SMILES CC1(C(N2CCC2n2cc(C3CCCOC3)nn2)=O)CCCC1(F)F N#CC1(C(N2CCCC(N3CCN(C(C4(O)CCCC4)=O)CC3)C2)=O)CCOC1 C1(C)(C(C)C)CN(C(=O)C=CCN(C)C(c2ccncc2F)=O)CCO1 N1(C(c2nc(C(C)OC)oc2)=O)CCC2(C1)CN(C(c1ccc(Cl)cn1)=O)C2 C1(CNC(c2nc(C)sc2)=O)CCC2(CN(C(c3ns[nH]c3=O)=O)C2)O1 c1(C(=O)NC(CSC)C(=O)O)cn(CCn2cc(C3COC3)nn2)c(C)cc1=O Cc1cc(NC(=O)C=CC(C)NC(c2c(C)cccc2O)=O)cc(Cl)c1 c1(OC)c(F)ccc(NC(N2CC(O)CC2CN)=O)c1F N1(C(C2N(CC#C)CCC2)=O)CCC(NC(c2c(C)cccc2Cl)=O)CC1C CCCC(C(=O)NCCC1CCC2CC12)NC(C1C=CCC1)=O C(=O)(C(C(C)C)OC(=O)C(F)C(=O)OCC)NC(C=C)COC C1(NC(C2C(C)CCC2)=O)CCCN(C(=O)C(C(C)O)N(C)C)C1 N1(C(c2cc(C#N)on2)=O)CC2(CCCC(CNC(C3CC(=O)N(O)C3)=O)O2)C1 C1(C(N2CCCC(N3CCCC3)C2)=O)CCCN(Cc2cccc(O)c2)C1 N1(C(C(CC=CC)C)=O)C2COCC1CC(NC(C1(C)CCNC1=O)=O)C2 C(=O)(C1=CCCO1)N1C(C(C)(C)CNC(=O)CC2CC2c2ccsc2)CCC1 c1(-c2cn(CC(=O)N(CC)Cc3cnn4c3NCC4)nn2)cc(F)c(C)cc1Cl C1(CC)(NCC(c2csc(=N)[nH]2)=O)CCCC1 c1(C2C(C(=O)NC3C(C=C)CC3)C2)cccc(Cl)c1Cl c1(C(N2CC(NC(C=CC)=O)C3C2C3)=O)cc(Cl)cnc1C CON(C)CC(O)C(=O)n1cc(-c2nc(CC3CC4CCC(C3)N4)cs2)nn1 C#CCC(C)C(=O)N1CCC(C)(NC(c2ncn(C(C)(C)C)n2)=O)C1 c1(C(=O)NCCN(C)C(C2CCCCC2C(C)(C)C)=O)ccncc1Br N1(C(c2ccnnc2)=O)CCN(C(C2(O)CCSC2)=O)CC1c1ccccc1 c1(C(N2CC(CCCNC(CCC(C)SC)=O)OCC2)=O)cc(O)ccc1Cl c1(C(N2CCC(O)(CCNC(c3cn(C)c(O)n3)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(CC)(NC(=O)NCc2cncc(-c3ccc(C)cc3)c2)CCCOC1 C1(CNC(CC(CC)C2CCC2)=O)CC2CCC1N(C(C1CC1C#N)=O)C2 c1(CNC(C(C)NC(c2n(CC=C)nnn2)c2ncsc2Br)=O)ccc(C)cc1 N1(C(N(C)Cc2cncnc2)=O)CCCC2NC(=O)C(C)(C)C12 C(=O)(CCCCC(F)(F)F)N(C)CC1CN(C(=O)CSCC2CCCO2)CCO1 C1(CNC(C(CC)(C)C)=O)CN(C(C2CN(CC(C)C)C2)=O)CC1(F)F C1(CNC(CSc2n(C)cnn2)=O)CC2CCCC2N1C(C1(CCN(C)C)CC1)=O N1(C(CCNC(=O)OC)=O)CC(NC(c2cc(C(F)F)nn2C)=O)C(C)C1 N1(C(CC2N(S(CC)(=O)=O)CCC2)=O)CCC(C)(CNC(c2ccsn2)=O)C1 N1(C(C2CC(CC)(CC)C2)=O)CCCC(C)(NC(C2C3CCCCCC23)=O)C1 c1(OC)cc(C(=O)N(C2CCC(NC(C3CN(C)C(=O)N3)=O)CC2)C)cc(Cl)n1 c1(C(N2CCCN(C(C3CCN(C)C3)=O)CCC2)=O)coc2c1C(=O)NCCC2 c1(C(=O)NC2C3CN(C(C(CSC)O)=O)C2C(O)C3)cnc2[nH]ccc2n1 c1(CC)oc(C(=O)NC2CCC(F)(CNC(C3(C=C)CCC3)=O)C2)cc1C c1(NC(=O)NC(CC(=O)OC)c2ccccc2)ccc(S(N)(=O)=O)cn1 c1(C(N2CCC(NC(c3cnc(SC)n3C)=O)C2C)=O)ccc2c(c1)COC2 c1(N(C)CC)ccc(N=c2c([N+](=O)[O-])c[nH]c3ccc(F)cc23)c(F)c1 N1(C(C(C)(C)CF)=O)CCC(C2CCN(C(c3ccco3)=O)CC2)C1 CCCCC(C)N=c1ccnc(NC(c2ccc(N(C)CC3CC3)cc2)C)[nH]1 c1(C(N2C(C(C)C)C(NC(=O)C(C)CF)CC2)=O)cnc(Cl)c(F)c1 N1(C(CN(CC(C)C)C(C2CCC(C)C2)=O)=O)CCC(CC2CC2)CC1 N1(C(C2(C#C)CC2)=O)C2CCC1C(C)C(NC(=O)Cn1ncnn1)C2 CC(CC(=O)N1CCN(C(=O)C=Cc2ccc(O)cc2)C(CO)C1)C(F)F C1(C(=O)NC2CCCN(C(C#CC(C)(C)C)=O)C2)Cc2ccncc2C1 C#Cc1cccc(NC(C(C)(C)c2ccccc2)c2nnnn2CC2CC2)c1 Cc1cc(C(=O)NC2CCCCC2NC(=O)Cc2ccccc2Cl)cn(C)c1=O C(CS(=O)(=O)CC(=O)N1CC(CNC(=O)C(F)C2CCC2)OC(C)(C)C1)OC CCCCC(C(=O)N(CCCO)CCC)NC(c1ccc(C(N)=O)[nH]1)=O N1(C(c2c(CC)noc2)=O)C2CCCC1CN(C(c1cccc(OC)c1Cl)=O)C2 C(C(=O)NC1CCN(C(=O)Cc2ccc(O)nc2)C1C)(C(C)C)NC(C)=O C(CCC(C(=O)Nc1cccc(Cl)c1C)N(C1COCC1n1ccnc1)C)OC N1(C(CC(=O)NCC)=O)CCC(C)C(NC(=O)CCCOCC)C1 C(CCCCC(=O)NCC1(O)CN(C(C)CC)C1)OCC.c1(C)ccc(CO)o1 CC1CC(CNC(=O)Cn2cnnc2)CN1C(C1CC(F)(F)CS1)=O N1(C(=O)COCc2ccccn2)CC2=C(C1)CN(C(C1CCCN1C(N)=O)=O)C2 N1(C(C)=O)CCCC1C(=O)NC1(CCNc2cc(C3CCC3)no2)CCCC1 Cc1cc(NC(=O)COC2CC2)cc(N)c1.N12CCN(CC1=O)C1CC(C1)C2=O C1(NCC(F)(F)F)(CN(C2CC2(Cl)Cl)C)CCCC1 C1(NC(C=C(C)C)=O)CC2CC(NC(=O)COCC3CCCO3)C1C2 N1(C(COC2(C)CN(C(=O)CS(N)(=O)=O)C2)=O)CCN2CCOCC2C1 C1(CCC(N2CC(COC)(CNC(c3csc(CO)n3)=O)C2)=O)CCC(O)CC1 CCC(C)(C#N)C(=O)N1CCC(O)(C(C)NC(c2nncnc2C(F)F)=O)CC1 C1(NC(C(CC)CC)=O)CCCN(C(=O)Cn2ccccc2=O)C1CC C(=O)(CCS(C)=O)NC(CC)CNC(c1ccc(OC)s1)=O C1(F)(CNC(C2CC23CC3)=O)CCCN(C(=O)C(F)(F)C2CCCC2)C1 Cc1cccc(C(O)C(=O)NCc2ccc(F)cc2C(F)(F)F)c1F C1(F)(CNC(=O)CCC2CC2(F)F)CCC(NC(c2cccnc2O)=O)C1 Cc1nn(C)c(F)c1C(N1CC(NC(c2scnc2C(C)(C)C)=O)CC(O)C1)=O N1(C(Cn2ccc(C)n2)=O)CC2CC(NC(C3(C4CCCO4)CC3)=O)C2C1 C(C(N=[N+]=[N-])C(=O)NCC(O)CNC(c1cnc(C(=O)OC)s1)=O)OCC C(CC(C(=O)NCc1ccc(C)cn1)NC(=O)Cc1cnc(C)n1C)=CC c1(C(C(=O)NC2(C)CC2)N(C(C(C)C2C(C)C2)=O)C)ccc(Br)c(F)c1 c1(C(N2CCN(C)CC2)C)nc(O)c2sccc2n1.c12ccccc1C(=O)N(C)C2 C#CC1CCN(C(C2C(NC(C3(SC)CC3)=O)C2(C)C)=O)C1 N1(C(C(CC#C)NC(c2oc(C)cc2C)=O)=O)CCC2(CCCOC2)C1 CCCC(C(=O)NC1CN(C(c2c(F)cncc2Br)=O)CC1C)S(N)(=O)=O Cc1cc(CC(=O)NCC2CN(C(C3C=CCC3)=O)CCO2)n(C)n1 C1(CNC(c2ncc3[nH]ncc3n2)=O)CN(C(=O)C2=CCC2)CC12CCOCC2 c12ccc(c(O)c1)CNC1CCCC1C(=O)N2.N1(CC)CCCCC1C#N N1(C(c2c(C)nc(CCC)o2)=O)CC2CCC1C2NC(c1coc(OC)n1)=O Nc1cc(Cl)c(Cl)cc1C(=O)N=c1cc(-c2cccc(F)c2)[nH][nH]1 N1(C(C2(OC)CCCSC2)=O)CCC(C2(NC(=O)C(C)C3CCC3)CCC2)CC1 N1(C(c2c(CC)cco2)=O)CCC(O)(CN(C(=O)C(C(F)(F)F)OC)C)CC1 c1(C(=O)NCC2CC(NC(C(n3ccc(C)n3)C)=O)C2)cc(F)c(C#N)c(F)c1 CC(C)(CCCCNC(=O)C(CC(C)(C)C)C(N)=O)C(=O)NNC(=O)c1ccon1 c1(CCOC)nc(=NC2CC(NC(=O)C=Cc3scnc3C)C2)s[nH]1 C1(C)(CNC(c2c(CC)occ2)=O)CC(F)(F)CN1C(=O)COCC1CCCC1 N=S(=O)(CCNC(=O)C(Cc1cccc(F)c1)C1CC1)c1ccccc1 O=C1CCN(C(=O)C(CCCl)C(=O)O)C(=O)c2ccc(F)cc21 c1(CC(C(=O)OC)Nc2cn(C)nn2)ccc(C=O)cc1.C(=O)(C1=CCSC1)N Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC1CC(O)CN(C(=O)C2=COCC2)C1 N1(C(CSCC(=O)OC)=O)CC(C)N(C(c2cc(C)n(C(C)(C)C)n2)=O)CC1C Cc1c(Cl)cc(C(=O)Nc2c[nH]nc2C(=O)NC(c2ccc(I)cc2)C)cc1Cl N1(C(C(COC)OC)=O)CCN(C(=O)C(C)c2ccsn2)CC1 C1(C)(CNC(C2C(C(=O)OC)CC2)=O)CCCN(C(C2NC(=O)OC2C)=O)C1 C(CCC1CC1)(C(=O)NOC1CCC(O)C1O)NC(C(CC=CC)C)=O C1(C(=O)OC(C)CC2CCC2)CCn2ccnc2C1 c1(C(CN(C(=O)NCC(C(F)(F)F)OC)C(n2ccnc2)=O)O)ccc(F)cc1F N1(C(COCC)=O)CC2COCC(C1)N2C(c1cccc(C#N)c1)=O N#Cc1ccc(C(=O)NC2CC23CCC(NC(=O)CC2C=CCC2)CC3)c(F)c1 c1(OCC(=O)OC)ccc(C(=O)NC2CN(C(=O)C=C(C)C(F)F)C2)cc1 C(=O)(C1CCc2nccn21)NCC1CCN(C(CCCOC(C)C)=O)C1 c1(OC)ccc(C(N2CCCC(O)(CCNC(C3CC(OC)C3)=O)C2)=O)cc1C Cc1ccc(Br)c(C(N2CCOC(C(=O)Nc3cscn3)C2)=O)c1F Cc1cc(-c2ocnc2C(=O)NCC2CCC2NC(=O)CCC2CCCC2)on1 CN1CCc2cc(C(N3CCC(CCNC(C4CC(C#N)C4)=O)C3)=O)sc2C1 C1(c2noc(C)n2)(OC)CCN(C(C2(C(CC(=O)OC)CC(=O)O)CC2)=O)C1 C1(C(=O)NCC(CCCC)NC(c2nnsc2SC)=O)C2CC3CC(C2)CC1C3 C12(CNC(C3CCCS(=O)(=O)C3)=O)CC(CO1)N(C(=O)Cn1ncnn1)C2 C1(CNC(CC(CC2CC2)NC(CC2C(CC)C2)=O)=O)CCCC2(CCC2)C1 C1(NC(CC2CC(OC)C2)=O)CCCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1C C1(NC(C=CCNC(COCCCC#C)=O)=O)CCn2ccnc2C1 N1(C(c2ccn(C)c2)C(=O)NC)CCCC2(C)CCCCC12 C12(CCCO1)C(=O)NC2.C(C(F)(F)Cl)NC(c1nncs1)=O C1(NC(C2(CCOC)CCC2)=O)CC2CC(NC(=O)CNS(C)(=O)=O)C1C2 C(=O)(C#CC1CCOCC1)N1CC(NC(COc2cccc(C)c2C)=O)C(C)C1 c1(N(C2CCC2)C)ncccc1S(=O)(=O)N(CCCCCCn1cnnn1)C N1(C(C(CC)CC)=O)CC2CCC(N=c3cc(Cl)nc(C4CC4)[nH]3)CC2C1 C1(CCNC(C(C)(C)OC)=O)CSCCN1C(=O)CSCC1CCOC1C(C)C C(C(C)C)(C(C(=O)NCCCF)N1CCCC(C)(O)CC1)OC N#Cc1cn(CC(N2CCCCC2CCNC(=O)CC(F)F)=O)c(=O)nc1O CCC(CNC(=O)Cc1c[nH]nc1C)(CC)C(=O)N(CCS(N)(=O)=O)C Cc1nn(C)c(C)c1C(C)C(=O)OC(c1ccccc1)Cc1ccc(F)cc1 c1(NCC2N(C(CCc3c(C)nn(C)c3)=O)CCC2)ccc(C(N)=O)cc1[N+](=O)[O-] CC1CN(C(=O)CC2CC2)CC1CNC(c1c[nH]nc1C1CCOCC1)=O C1(NC(c2ccnc(OC)n2)=O)CCN(C(c2c(Cl)csc2Cl)=O)CC1O N1(C(c2cc(CC)nc(Br)c2)C(=O)NCCCC2CC2)CC(CO)C2(CCC2)C1 C=CCC(C)(C)CC(=O)N1CC2CC(NC(=O)CC3CCCNC(=O)C3)C2C1 C1(NC(Cc2scc(CC)n2)=O)CC2C1CCN2C(=O)CC(C)C(C)C c1(C(=O)NCC2N(C(C=COCC)=O)CCC2)c(C)cc(O)cc1C N1(C(C2(OC(C)=O)CC2)=O)CCC2CC2(C(=O)NC2CN(C)CC2(C)C)CC1 C1(C(=O)NCc2scc(CNC(C3C(C)(C)C3)=O)n2)CC2CCCCCCC12 N1(C(C(=O)OC)=O)CC2CC(C)N(CC3CCNC4(CCC4)C3)C2C1 C1(CC)CCN(C(=O)C(CN(C)C)SC)C1C(=O)NCCCN(C)C(C)C c1(CC(N2CCC(C#N)(c3cc(F)cc(F)c3)CC2)=O)csc2ccc(Cl)cc12 CC1C(NC(=O)CCC[N+](=O)[O-])CC2CCC1N2C(c1cnoc1C1CC1)=O C(=O)(C1=CCC(C)(C)CC1)N1CC2C(NC(CCNC(=O)OCC)=O)C(C2)C1 c1(C(N2CC3C(CNC(C)C)C3C2)=O)c(F)cc(Br)cc1F C1(N(C)C(c2ncn(C)n2)=O)CN(C(c2cc(Br)cnc2S)=O)CC12CC2 C(CC1CC1)(C(=O)N=c1cc(C)n(C2CC2)[nH]1)C(C1CN(C(C)=O)C1)=O C1(OC)(CNc2ccc(F)cc2CNC(=O)OC)CC(C)CC(C)C1 c1(C(=O)NCC(N(C(C(CCC)OC)=O)C)C2CC2)nc(N)cc2ccccc12 C1=CC(N=c2[nH]c(=NCc3nccn3C3CC3)[nH]c3c2CCCC3)CCC1 c1(CNC(c2ccc(C(C)=O)[nH]2)=O)ncc(C(=O)NCCC(O)CC2CC2)cn1 C1(NC(CCCCC)c2nnnn2C2CCOCC2)CCc2nncn2C1 C1(C(=O)NCCn2cc(-c3csc(C4CC4)n3)nn2)CCC(F)(F)CC1 N1(C(C(CC)(C)O)=O)CCN(Cc2nc(-c3ccccc3)no2)C(C(F)(F)F)C1 Cc1cc(C(=O)NC2CCCC(CCNC(c3ocnc3C(F)F)=O)C2)nn1C C1(C(=O)NC2C(SC)COC2)COCCC1NC(C1CC=CC1)=O c1(CC(=O)N(CC(C)O)CCNC(C2(F)CC2C)=O)nccn1C C1(CC(=O)N(CC#C)CC)CN(C(=O)C(C)N(C)C(C)=O)CCC1C Cc1cc(C(N2CCC(C)C(CC(=O)NCc3ccccc3Cl)C2)=O)nc(C)n1 C#Cc1cn(C)nc1C(N1C2CCC1C(NC(=O)Cn1cc(C(C)O)nn1)C2)=O c1(C(=O)NC2C(CNC(=O)C(=O)NCC(F)(F)F)C2)cc(Cl)c(F)cc1F CCCCC(C(=O)N1CCCCC(Cn2cc(C3(O)CCCC3)nn2)C1)OC N1(C(C(CC)OC2CCCC2)=O)CC2CC2(CNC(c2cccnc2S)=O)C1 C1(C(C)(C)C)(CNC(C2CC(CO)C2)=O)CCCN1CC.C(=O)(C(=O)N)NCC1CC1 C(=O)(C(C)CC(F)(F)F)NC1CC(C(=O)NC2(C(N(OC)C)=O)CC2)C12CCC2 c1(C(=O)NCCN(C(=O)C(O)Cc2cc(Cl)cc(Cl)c2)C)coc(S(C)(=O)=O)c1 C(=O)(CCCCC(F)(F)F)N1CC(C2CN(C(C3(CC#C)CCCCO3)=O)C2)C1 Cc1cnn(C)c1CC(=O)NC1CCCC1NC(=O)CN(C)Cc1ccccc1 c1(C(=O)NC2CC(CNC(CC3C(C)(C)OCC3)=O)C2)ccc([N+](=O)[O-])o1 c1(C(N(C2CCN(C(c3csc(C)c3)=O)CC2)CC#C)=O)cncc(F)c1 Cc1cc(C(N2CCC(C)C(N(C)C(c3cn(C)c(C)n3)=O)C2)=O)c(C)c(C)c1 N1(C(c2nc(C)n(C)n2)=O)CC2(CC(NC(=O)COCC(C)(C)C)CO2)C1 CCCC(C(F)(F)F)NC(C1(CF)CCN(C(C2CC3(CC3)CO2)=O)C1)=O C1(CNC(C(C)Cc2ccco2)=O)CCC(C(=O)N(C)CCF)CC1 c1(C(C(=O)NCC2CCCO2)N(CC(=O)NCCC)C)cc(CC(C)C)on1 C1(C(N(C(c2ccc(OC)cc2)C(=O)O)C)=O)Cc2cc(C)ccc2S1 c1(C(=O)NC2(CO)CCN(C(C3C4CCC3CC4)=O)CC2)cncc2nc[nH]c12 c1(CN(CCCOC)C)csc2c1CCC(C)C2.N12CC(O)(C1)CNC2=O c1(NC(C2CC(F)CN2Cc2c(O)cccc2Br)=O)ccn2ncnc2c1 CCC(CC)CCCNC(=O)CC(C)CNC(C1(C)CC2C=CC1C2)=O O=C(CCC(F)(F)F)NCC(c1ccccc1)NC(C1CCCS1(=O)=O)=O C1(CNC(CCC(C)(C)OC)=O)CCN(C(=O)CCC(C)(C)C#N)CCC1(F)F C(C1=NOC2CCCC12)NC(c1ncc(C)c(C)c1)=O CC(C1CCCCC1)=CC(=O)NC1CCCC1CNC(=O)C1=CCCC1 Cc1cc(=O)c(C(N2CC(N(C)C(C34CCCC3C4)=O)C(O)C2)=O)cn1C N1(C(c2ccc(NC(C)(C)C)cc2)=O)CCC2(NC(C3CC3F)=O)CCCC12 C1(c2nc(C)[nH]n2)CCN(C(c2ccccc2)=O)CC1.C12CCN(C1)OC2=O CN1Cc2cc(CNC(=O)COc3ccc(Cl)cc3)ccc2C1=O C1(NC(CCCC=C)=O)CCN(C(C2(C(=O)N(C)C)CC2)=O)CC(C)(C)C1 N1(C(Cc2c(C)nsc2)=O)CC2CN(C(=O)CNC(=O)Cn3cncn3)CCC12 N1(C(C(C=C)O)=O)CCC(NC(=O)CCCN(C)C(C)C)C(CO)C1 CCC(C)CC(C)Nc1cncc(-n2cc(CN(C)C)nn2)n1 C1(NC(CSCCC)=O)CCCC(NC(C2COCCOC2)=O)C1 C1(=CC(=O)NC2CC(NC(C3C(C)(C)C3)=O)C2)CN2CCC1CC2 CC1(C)CC(NC(=O)CCc2ncc[nH]2)CCN(C(C2(C#N)CCOC2)=O)C1 c1(OC)ccnc(CNC(C2CC3CCCC23)=O)c1OC CCC(CC(=O)NC1(CCOC)CCN(C(c2c(C)ncn2O)=O)C1)C(F)F C(=O)(C(C(C)C)n1ccc(C)c1)NC(C1(OCC)CCC1)(c1nn[nH]n1)C c1(C(N2CCC(NC(CC#C)=O)C2)=O)ccc(F)c(I)c1 C(=O)(C1(C)C(=O)O1)NCC(CO)NC(CC)=O.C(C)(C)(C)OC(C)=O.OCC CC(C)(C)C(C#N)C(=O)N1CC(O)(CC2CC2NC(=O)CCCCc2cnc[nH]2)C1 C1(NC(=O)CCOCC(F)F)COC2(CCN(C(=O)CSC(F)F)CC2)C1 c1(C(=O)NC2CC(C)N(C(c3c[nH]c(=O)cn3)=O)CC2)ccc(F)c(F)c1F C(=O)(C1=Cc2ccccc2C1)N1CCC(C)CC1C(N1CCN(C)C(CO)C1)=O N1(C(C23C(NC(C(C)=CC=C)=O)C4CC2C3C4)=O)CCCC2C(=O)NCC12 CC1=C(C(=O)NC2CC3CCC2C(NC(c2cnnn2C(C)C)=O)C3)CCCO1 c1(OC)cc(OC)ncc1C(N1CC(C(=O)O)C(C)(C)C1)=O CC(C)(O)CCCC(=O)N1CC(CNC(c2cncc(O)c2)=O)C1 c1(CCC)cccc(C(=O)N(CCNC(c2cc(C(F)(F)F)n[nH]2)=O)CC)c1 N1(C(C)=O)CCN(C(C2C3COCC23)C(=O)NCCC2CCCOC2)CC1 C1(C(C(=O)NCC2(NC(=O)C=Cc3ccccc3)CCOC2)=O)CCCOCC1 N1(C(C2C(C(=O)OC)C2)=O)CCCCC1CN(C(=O)CC1CC2(CCC2)C1)C N1(CC(C(=O)NCc2c(C(=O)OC)ncs2)OC(=O)NC(C)(C)C)CCCCCC1 C12(C(=O)NC3C=CCN(C(c4cc(C)n(C)c4)=O)C3)CCCC1C2(F)F c1(SC)ccc(C=CC(=O)NCC2(OC)CN(C(C3CC3C)=O)C2)cc1 C(C)(CC(C)NC(=O)CC(C)O)NC(C=C(C)CN1CCCC1)=O C1(NC(CCSCC)=O)CCN(C2CC2)C1 c1(NC(Cn2cc(C(CCC)=O)nn2)=O)coc(S(C)(=O)=O)c1 c1(OC(C(=O)NCCN(C(C2N(C(C(C)C)=O)CCC2)=O)C)C)cccc(F)c1 N1(C(C(C2CC2)NC(c2cc(Cl)cs2)=O)=O)CCCC2(CC1)CC2 Cc1cc(C(N2CSCC2C(=O)Nn2cnnc2C)=O)cc(C#N)c1 C1(COC)CN(C(c2cc(C)[nH]n2)C(=O)NCCC2(C)CC2)CC1C c1(CC(=O)NCCN(C(=O)CCC=C(C)C)CCOC)ccc(OC)nc1 CCCC(C(O)C(=O)N(C1CCOCC1OC)C)NC(=O)C1CC1 c1(COCCC2(C(=O)NC3CCN(C(=O)C(O)CF)C3)CC2)cccc(Cl)c1 c1(C(=O)NCCC2C=CCC2)ccoc1CNC(C1CC1(F)F)=O C1(CN(C)C(C2CC(=O)N(C)C2)=O)CN(C(=O)C=C(Cl)Cl)CCO1 C(C(O)CC(F)(F)F)NC(CC1CCC(NC(C2(C)CC2(F)F)=O)CC1)=O C=CCCCCC(=O)NCC(N1CCN(C(C2CC2C2CC2)=O)CC1)=O C#CC1(C(=O)NCC(O)CCC2CC2)CN(C(=O)C(O)CC=C)C1 c1(OC)cccc(N(C(=O)Cc2ccns2)C)c1.c12nc(co1)C(=O)NC2 c1(CNCc2ccc(C)nc2)cc2cccc(Cl)c2s1 N1(C(C(C2CCOCC2)OC)=O)CCC(N(CCO)C(C2CC(F)(F)C2)=O)CC1 C12(CNC(C(C=C)OC)=O)CCC(C1)N(C(c1sc(F)cc1C)=O)C2 C(N=c1[nH]c2ccc(Br)cc2s1)C1CC(C)N(C(c2cccc(C3CC3)c2)=O)C1 CC1CCCCC1(CNC(=O)Cn1ccc(O)nc1=O)NC(=O)Cc1cnsc1 c1(CCC(=O)NC2CCN(C(CSCC=C)=O)C2CC)cc(F)ccc1F Fc1ccc(CC(F)CNc2cccc(C(F)(F)F)c2)cc1F c1(C2C(NC(C(CNC(c3cc(COCC)[nH]n3)=O)C)=O)C2)ccccc1C C1(CCNC(c2c(CC)cco2)=O)CCN(C(C2CC(N(C)C)C2)=O)C(C)C1 C12(CNC(CC3CC(OC)C3)=O)CCC1CN(C(c1ccnc(F)c1N)=O)C2 N1(C(c2cn(CC3OCC(C(=O)OC)C3)nn2)=O)CC(C(N)=O)CC(C)C1 Cc1c(C(N2CCC3S(=O)(=O)OCC3C2)=O)c2ccccc2n(C)c1=O c1(C2(C(=O)NC3(CNC(C4CC5CC5C4)=O)CCCC3)CCCC2)ccc(Cl)cc1 C1(NC(C(CC)C(C)C)=O)CC2CCCC(C1)N2C(c1nnsc1C)=O N1(C(C2C=C(C)CS2)=O)CCCC(C)(C)C1C(=O)NC1CCC1 C1(NC(=O)OC(C)(C)C)CC2CCC1N(C(=O)CC1CCC3CCCCC3C1)C2 C(CCCCC(=O)NC1CC(CN(C)C)C1)OCC.C12(C)CCC(CC1)NC2=O c1(C(N2C(CCNC(c3csc(C)c3N)=O)CCC2)=O)nc2c(s1)CN(C)CC2 Cc1nn(C)c(C(N2CCCC(CCNC(=O)CC3COCCO3)C2)=O)c1Cl c1(C(=O)NCCc2ccc(OCCCC)cc2)ccc(F)c(Cl)c1 C(=O)(C(C(C)NC(=O)COCCF)C(C)C)NCC(C)N(C)C1CC1 Cc1nn(C(C)C)cc1C(=O)NC1CCCC(NC(=O)Cc2ncn(C)c2C)C1 C#CC1(C(=O)NC(CC(=C)C)C2CC2)CCN(C(c2cc(Cl)c[nH]2)=O)C1 C1(CC(=O)NCC(CC)C)CN(C(C2CC(=O)CC(=O)N2)=O)CC12CC2 c1(C(=O)OC)cc(C)ccc1S(=O)(=O)N(C1CCCCC1N)C C(=O)(C(C(C)C)N1CCC(C)CC1)NC1(C)CN(C(CCc2nnc(C)o2)=O)C1 c1(N2CC(C)(C(F)F)OCC2)nc(N2CCOC3(CCCC3)C2)nc2sccc12 c1(C(=O)NC2CC(NC(=O)CC(O)CC3CC3)C2)cnc(O)c2c1NCCC2 N1(C(CCN(C(C(CC(CC)C)=O)=O)CCO)=O)CC2C3C=CC(C3)C2C1 C1(C(N(C)CC2CCN(C(C3(Cl)C(C(C)=O)C3)=O)CC2)=O)CN2CCC1(C)CC2 CC(C)(CC(F)F)C(=O)N1CCC(O)C(NC(C2CCC=CCCC2)=O)C1 C1(C(=O)NCC(CNC(c2conc2-c2ccccc2)=O)O)CCC(CO)CC1 c1(C(N2CCC(C=C)(CO)CC2)=O)ccc2cc(C)oc2c1 C1(NC(C2CC3C=CC2C3)=O)CN(C(=O)C2=CCCCO2)CC12CCOCC2 Cn1cc(C=CC(N2CCC(OCC(N3CC(CC(F)F)C3)=O)C2)=O)cn1 Cc1nc(S(C)(=O)=O)ccc1N(C1CCNCC12CC2)C(=O)C(C)CN c1(NC(N2CC(F)(c3ccccc3)C2)=O)c(F)cc(F)cc1F c1(C(=O)NCC23C(CN(C(C(ON=C(C)C)C)=O)C2)C3)n[nH]c2c1CCC2C N1(C(C(C)OCCN(C)C)=O)CC2(C1)CN(C(C1CC(F)(CO)C1)=O)CCO2 C1(COC)CCCN(C(=O)NC(c2ccc(OC(F)F)cc2)C)CC1 CN1C(=O)CCCC1C(N1CCC(n2cc(CNC(C3CCCO3)=O)nn2)C1)=O C(=O)(C(C(CC)CC)OC)NCC1N(C(c2c(Cl)cn(CC)n2)=O)CCCC1C C(=O)(C1=CC2CCCC12)N1CCCC(CNC(c2c(C)cc(C)o2)=O)CC1 CS(=O)(=O)c1cc([N+](=O)[O-])ccc1N.C12(C(N)=O)CC3CC(C(=O)N1)C2C3 C1(O)(CN(C(=O)C=CCN2CCCC2)C)CCCN(C(C2(CO)CCOC2)=O)C1 N1(C(C2(C#N)CC3CC3C2)=O)CCCC12CCCN(C(c1scnc1Cl)=O)C2 C(CCC(=O)NCC1(NC(c2cnco2)=O)CC1)OCC(C)C c1(CNCC(CC)Oc2ccccc2)csc2ccc(C(=O)O)cc12.N(C)(C)CN CCCCC(CNC(=O)Cc1nccn1CC)NC(c1cc(CC(C)C)on1)=O N1(C(c2n(C)cnc2)=O)CC(C)(C)C1Cn1cc(CS(C)(=O)=O)nn1 N1(C(C(C)(C)C)=O)CCN(C(=O)CCOCC(F)(F)C(F)F)C2CC12 c1(SCC)ccc(C(=O)NC2CCCC2NC(C2CCOC2C2CC2)=O)cn1 c1(C(N2CCN(C(C3(CC)CCNC3=O)=O)CC2)=O)ccc(=O)n(C)n1 c1(CN(C2C(C)CCNCC2)C(c2cccnc2)C)cc(S(N)(=O)=O)co1 C(=O)(CC1CCCc2ccccc21)N(C(CNC(CC(C)CF)=O)C)C N1(C(CCN(C(=O)CCC2CCCOC2)CCCO)=O)CCOCC2(CC2)C1 C1(C(N2CCC(NC(C(CC)(F)C(=O)OC)=O)CC2)=O)Cc2ccc(F)cc2C1 C(=O)(CCCC(C)(C)CC)N1CCCC(N(C(c2cc(CC)cc(C)c2)=O)C)C1 c1(C(=O)NCC(C)(C)CNC(c2occc2C2CC2)=O)c[nH]c2nc(Cl)ccc12 c1(C(=O)NCC2CC(NC(CC3(C=C)CCC3)=O)C2)cc(Cl)c2c(c1)OCCO2 C1(C(=O)NC(c2cccnc2)c2nn[nH]n2)CCc2ccccc2C1 C#CCC(C(=O)N(CC(C)(C)N(C)C)C)NC(c1cc(C)oc1C)=O C1(NC(CCc2onc(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(O)C1 Cc1cc(Cl)c(C(=O)NC(C)CCCNC(c2cc(C(N)=O)no2)=O)cc1C C=C(C)C(CC(=O)NC1CC1NC(=O)CNS(C)(=O)=O)OCC C1(NC(C2CCC(C)CC2)=O)CC2CCC(C1C)N2C(C1(C)CCCS1(=O)=O)=O c1(C(=O)NCC2(O)CCN(C(C3C(CC)C3)=O)CC2)ccnc2c1CCO2 CCCC(C(O)C(=O)N1CC(CO)C(C)C1)NC(=O)C(F)=C(C)C N1(c2c(C)cnc(-c3c(SC)ccnc3)n2)CCCC2(CNC(=O)O2)C1 CC(C)CC(O)CC(=O)N(C1CCN(C(=O)CC(F)(F)Cl)CC1C)C Cc1cccc2cc(C(=O)NC(c3ccc(C(=O)O)c(C)c3)C)sc12 N1(C(C(C)CF)=O)CCCC(Cn2cc(CC3NCC3)nn2)C1.N1CCOC1=O Cn1cc(CC(=O)NC2CC2CNC(=O)Cn2cc(C3CC3)cn2)c(Cl)n1 N1(C(CC(CNC(C(C(CC)C)N(C)C)=O)C2CCC2)=O)CCC(N=[N+]=[N-])CC1 CC(CC(C)NC(=O)C=CC(C)(C)C)NC(=O)CSCC(N1CCCC1)C C1(NC(C2N(C(CC(C(C)C)C)=O)CC=C2)=O)CCN(C)CC1(C)C NS(=O)(=O)c1csc(C(=O)NC(C2CCOC2)CNC(c2ccnnc2O)=O)c1 C1(OC)CN(C(C2CC(F)(F)C2)=O)CC1NC(C1(c2cccnc2)CC1)=O C1(NC(C=C(C)C(F)F)=O)CN(C(c2nnn(C(C)(C)C)n2)=O)CC12CCC2 c1(C(N2CCN(C(C3OCC4CCC3C4)=O)C3(CC3)C2)=O)ccc2nc(S)oc2c1 Cc1ccc(C(=O)NC2CCCCC2CNC(=O)CC(O)CN(C)C)cn1 CC(CN=c1[nH]c2ccc(F)cc2s1)N(C(=O)CC1CC2(CCC2)C1)C c1(N(C(=O)CC2CCCN(C(=O)C(c3ccccc3)=O)C2)C)ccc(Cl)c(F)c1 c1(N(C)C)cc(C(=O)NCC2CCC(NC(C3C4CCOCC34)=O)CC2)ccn1 CCCCC(O)CC(=O)NC(CCOCCO)C(N1CCC12CCCCC2)=O n1(CC)nc(C2CC2)cc1C(N1CCC(C)C1CNC(=O)C(C)c1cncs1)=O C1(C(=O)NCC2(CNC(=O)CSc3n[nH]c(O)n3)CC2)(OC)CC(C)CC(C)C1 CN1N=C(CC(=O)N2CC3CC2C3CNC(c2ccc(C(N)=O)[nH]2)=O)CC1=O c12cc(ccc1F)C(=O)N2.N1(C(=O)NC(CN2C(C)CC2)C)CCOCC1 c1(NC(c2c(CNC(c3cccc(NC)c3)=O)c[nH]n2)=O)cc(F)ccc1O c1(OC)ccc2[nH]c(C(=O)NCCCNC(=O)CC3CCC3)cc2c1Cl CCC1=C(C(=O)NCC2CC(NC(c3oc(CC)nc3C)=O)C2)CCCO1 C1(NC(Cc2cc(C)sc2)=O)CN(C(C2CCCN2CC(F)(F)F)=O)CC1(C)C N1(C(C(Cc2ccoc2)NC(C2C(C)=CCS2)=O)=O)CCn2ncc(C)c2C1 C1(CNC(=O)COc2cccnc2)CC2CCC1N2C(c1ncc(Cl)cc1F)=O Cc1cc(C(N2CC(C3(NC(=O)C=Cc4ccccc4)CC3)C2)=O)cnc1O C(=O)(C1=CC2(CCN(C(C3CCCCC3)=O)C2)C1)NCCC1C(C)(C)CCC1 c1(C(=O)NC(CNC(c2c(C)[nH]c(C)c2C)=O)C)cc(Cl)cc(Cl)c1F C1(C)(C(=O)NCC(C)CN(C)C(c2cc(C(F)F)n(C)n2)=O)CCC12CCC2 CCCCCC(O)C(C)C(=O)NCCN(C)C(c1ccc(C(C)C)o1)=O c1(C(=O)OC)cnc(C)nc1N(C1CCCN(C(=O)CCC(F)(F)F)C1)C C(=O)(CCCCN(C)C)NC(C(=O)NC(C1CN(C)CCO1)C)CN(C)C C1(CNC(C(C)=O)=O)CC2(CCN(C(c3cccc(F)c3F)=O)CC2)CO1 N1(C(C2(NC(CSCC)=O)CCCC2C)=O)CCC2C(O)CC12 Cc1cc(-c2nc(-c3occc3F)n(C3CCCC3)n2)c(C)o1 C1(NC(C(C)c2ccco2)=O)CC2(CCN(C(C3C4CCCCCC34)=O)CC2)C1 C1(NC(COC2CCN(C(COC3(C)CCCC3)=O)C2)=O)CC1C1CC(F)(F)C1 C(=O)(C(Cc1ccccc1)CCS(C)(=O)=O)OC(CCCC)C O=C(NN1CCCOC1=O)C(CCc1ccccc1)NCCOCCO c1(C(=O)NC2C(C=C)CN(C(=O)C(C)S(C)(=O)=O)C2)nc2cnccc2s1 N1(SCCNC(c2occ(C(=O)OC)c2)=O)CCC2CCCCC2C1 c1(CNC(C2CC2C(F)(F)F)=O)ccc(-n2cc(C3CCOCC3)nn2)cc1 C(=O)(CCC(O)C(C)(C)C)OC(C#CCOC)OC N1(Cc2c(Br)c(C)n(C)n2)CC2C(C1C(=O)NCC1NC(=O)NC1=O)C2(C)C N1(CC)C(=O)CCC1C(=O)N(CCCNC(C1CC1c1ccncc1)=O)C(C)C CCC(COC)S(=O)(=O)N(CCN1CCCC1)NC(C)=O c1(C(=O)NCC2(CNC(C3CC(C)(F)C3)=O)CCCCC2)ccc(Cl)cc1F C1(C(=O)NC(C)CCNC(c2cc[n+]([O-])cc2)=O)CCCCS1(=O)=O N1(C(c2ccc(C(=O)NC3CC(C#N)C3)o2)=O)CCCC2CCCC12 N1(C(c2c(C)c[nH]c2)=O)CC(C(=O)N(C2CC(F)(F)C2)C)CC(C)(C)C1 N1(C(C(CSC)OC)=O)CCC2CCCC(C1)N2C(c1cc(N)cc(O)c1)=O C1(O)(C(C)NC(C2C=CCCC2)=O)CCN(C(c2csc(Cl)n2)=O)CC1 C(=O)(C1CCc2c[nH]nc21)OCC(C)(C)C.C123CCC(C1C2)ONC(=O)N(C)C3C CC1CCN(CC(N2CC(NC(c3cc(C(C)C)on3)=O)C2)=O)CC1 CN=c1ccc(C(N2CC=CC2CNC(C2(SC)CC2)=O)=O)c[nH]1 N1(C(C2CC(C)N2C(=O)Cc2ccco2)=O)CC2(CCC2O)C1 CC(CC(=O)NCC1CCN(C(c2cnn(CCN(C)C)c2)=O)C1)C1CC1 Cc1nn(CC2CC2)c(C)c1CC(=O)NCC(C)NC(c1nn(C)cc1Cl)=O C1(CNC2CCCN(C(c3scc(C)c3)=O)C2)COc2ccccc2O1 N1(C(CCCC#N)=O)CCCC2(C1)CN(C(c1ccc3cccnn13)=O)CCO2 C1(CNC(CC2CCCC(C)O2)=O)CCCCCN1C(=O)CCN1CCCC1 CS(=O)(=O)c1cccc(-n2cc(CONC(c3ccc(Br)cn3)=O)nn2)c1 n1(CC)ncc(C(=O)NC2CCCC2NC(=O)COCP(C)(C)=O)c1C1CC1 C(=O)(C(C(C)(C)C)OC)N(CCCCCC)CCNC(c1sc(C)nc1C)=O c1(OC(C)(C)C)ccc(COC(F)(F)F)cc1.c1(C(C)NCN)ccncc1 N1(C(CC(C)N2CCCC2=O)=O)CC(CNC(c2ccc(Cl)[nH]2)=O)CC1(C)C C1(NC(c2cncc(OC)c2)=O)CCN(C(c2cc(OC)ccc2O)=O)CC1O C(C)(C)(C#CCCCC)NC(C1C(C=CC)CN(C(=O)CC(O)CC)C1)=O C1(CNC(CCCN(C)C)=O)CN(C(c2cc(C3CCC3)no2)=O)CCC1(F)F CC1CC(C(=O)NC23CCC(C(=O)O)(CC2)C3)CC(C)S1(=O)=O C(CC(C(C)C)NC(c1ccc(OC(F)(F)Cl)cc1)=O)N(C(C1C(=C)CC1)=O)C C=C(Cl)CC(C(=O)N1CCC1C(N)=O)NC(=O)C(n1nccc1C)C c1(C(=O)NC(CSC)(C)C(=O)NCC(C)(C)N(C)C)cc(N)cc(F)c1 N1(C(C(C)(C)C2CCC2)=O)CCC(OC(F)F)(NC(=O)CSC(F)F)C1 c12cn3c(n1)CN(CC3)C2=O.c1(Nc2ccnc(OC)n2)ccc(Br)c(C)n1 N1(C(=O)C(c2ccccc2)O)CCN(C(c2ccnn2C2CCC2)=O)C(CO)C1 Cc1ccc2c(c1)CCC2Nc1cc(C(F)(F)F)ncn1.n12c(=O)nc([nH]1)N=N2 N1(c2ccnc(NC3(c4ccc(CO)cc4)CC3)n2)CCC2(CCSCC2)CC1 C12(C(N(C(C)CCNC(C3(C(F)(F)F)CC3)=O)C)=O)CCC(CC1)C2(C)C CCC(CC(F)F)C(=O)NC1CN(C(=O)Cc2ccccc2F)CCC1(C)C C1(NC(C2C(C(N)=O)C2)=O)C2CC(O)C1N(C(C1CCC3(CC1)CC3)=O)C2 Cc1ccc2c(c1C(=O)Nc1ccccc1CN)CCCN2 C1(OCCONC(=O)C2(C(C)OCC(C)(C)C)CC2)CCC(=O)NC1 N1(C(CC(C)C(F)(F)F)=O)CCC2CCN(C(=O)C3=CCCCC3)C2C1 C(C(CC(F)(F)F)NC(=O)CCc1conc1C)NC(C1CN(CC)C(=O)C1)=O CN1CC=C(CC(=O)NCCCCC2CCCN(C(=O)C=CCO)C2)CC1 c1(C(N(C2CCN(C(=O)CN3CCC3C)C2)CC)=O)cc(C(F)(F)F)nn1C CN1CC(NC(N2CCS(=O)(=O)CC2c2ccccc2)=O)CC(F)(F)C1 C1(NC(C2C(=C)C2)=O)CCCN(C(=O)CN2CCCC2=O)C1CC OC1CN(Cc2ccc(C3CCOC3)cc2)CCC12CCOCC2 N1(C(c2cc(CNC(C3CCCSC3)=O)on2)=O)CC(F)(F)C(F)(F)C1 C1(CC(=O)NC(CNC(CC(=O)NCC#C)=O)CC)CCC2CC1C2(C)C C(CC1=CCN(C(=O)CCc2ccsc2)CC1)NC(C12CCC(C)(C1)CO2)=O CC(C(C(=O)NC1CC1)N(CCCSC(F)F)C)C1(C)CC1 C1(C(NOC)=O)CCN(C(=O)CC2CC(C)=NO2)O1 N1(C(C2C(C)(C)C2)=O)CCCC2CN(C(c3cnnn3C3CC3)=O)CCC12 CCC(CC(=O)N1CCC(NC(=O)CCc2cncnc2)C12CCC2)C(C)C CC1(C)CC(NC(=O)COC(F)(F)F)CCN(C(C23CC(C(F)F)(CO2)C3)=O)C1 c1(C(=O)NCC(C)(C)NC(C(CC=CCC)C)=O)ccn2cnc(C)c2c1 C1(C)(C(=O)NCCC2CCN(C(COCCCOC)=O)C2)CC(C)(C)OC1=O N1(C(C(C2CCOC2)NC(C(CC#C)O)=O)=O)CC(C2CC2)(CO)C1 N1(C(CC)C)CCC(N=c2cc(C)nc(N(CCN3CCCCC3)CC)[nH]2)C1 c1(NCC(CC(C)C)C)ncc(-c2ccccc2)cc1F CCC(CCOC)C(=O)N(CC(=O)OC)Cc1cn(-c2ccc(CC)cc2)nn1 C(=O)(CC(C)(C)CC(F)(F)F)N1CC2(OCC(NC(C3CC(OCC)C3)=O)C2)C1 c1(-c2nn(CCCS(C)(=O)=O)c(C3CCOC(C(=O)O)C3)n2)cc(F)cc(F)c1 N1(C(c2cc(O)nc(O)n2)=O)CCC2CN(C(C3CCCC(O)C3)=O)C2C1 c1(CC(=O)NCC(CNC(=O)C(C2CCCO2)C2CC2)O)ccnnc1O Nc1cc(C(N2CCC(NC(c3cc4occc4s3)=O)C(O)C2)=O)cc(O)c1Cl N1(C(C(n2ccc(C)n2)C)=O)CCCCC(NC(c2cc(C(F)(F)F)ns2)=O)C1 C12(COC)COC(C(=O)NC3CCN(C(c4csc(COC)n4)=O)C3)(C1)C2 n1(CC)nnc2c(N3CC4(CN(C(C5(CCF)CC5)=O)C4)C3)ncnc12 N1(S(c2c(C(=O)O)cccc2)(=O)=O)CCC2(CC1)CC2NCCc1ccccc1 C(=O)(C#CC1CCOC1)NC1C(CC(=O)N(CC(CC)O)CC)C(O)C1 c1(C(=O)NCC(CO)NC(c2cnc(CC)s2)=O)ccc(C2CC2)nc1 Cc1cc(Cl)ccc1OC(F)F.C1(N(C(CO)=O)CCO)CCCN(C(=O)CO)C1 c1(C(N(C2CCN(C(=O)CS(=O)CC)CC2)CC)=O)cc2ccc(C)n2cn1 c1(C(=O)NC(CCN(C(c2cc(C)c(C)o2)=O)C)C)csc2c1CCCC2 c1(C(N(CC(C)NC(C2(COC)CC=CC2)=O)C)=O)cn2ccnc2cn1 c1(CC(=O)NC(c2c(C)nco2)=O)cccc(NC(C2(C(=O)NC3CC3)CC2)=O)c1 c1(C(C(=O)NC(N(C(C)CSCc2ccccc2)C)=O)O)ccc(F)c(F)c1 C1(OC)CC(NC(=O)CC2(C)CC(F)(F)C2)C12CCN(C(c1ccco1)=O)CC2 C(=O)(C1=NOC(C(=O)NC2(c3ccccc3)CC2)C1)N(CC(C)N)C.CS C1(C(C)NC(c2ccn(CC)n2)=O)CCN(C(=O)C(c2cscn2)N(C)C)CC1 CC1CN(C(=O)C=CC=C(Cl)Cl)CC(C)(C(F)F)O1 c1(C(=O)NCCN(C(=O)C(C)(C2CC2)OC)CC)cccc(N(C)C)c1 C1(c2nnnn2C2COC2)(NCCCOCC(F)(F)F)CCN2CCC1C2 c1(C(=O)OC)ccc(C(CC(=O)O)N(CCCS(C)=O)C)cc1 c1(C(N2CC(CCNC(CN(CCCCCC)C)=O)C2)=O)cnc(Cl)c(N)c1 Cn1nc(Cl)c(C(=O)NC2CCCN(C(c3ccc(C(C)(F)F)cc3)=O)C2)c1Cl N1(C(C(CC(C)C)C)=O)CCC2(C1)CN(C(c1cc3nccnc3[nH]1)=O)C2 C(CN=c1cc(C2CC2)nc[nH]1)COc1ccc(Cn2ncc(N=[N+]=[N-])c2)cc1 c1(C(=O)NCC(C2CCN(C(CC(CC)C)=O)CC2)F)ccc(Cl)c(N)c1 Cc1ccc(CS(N2CCOC(CCC(=O)NC3CC3)C2)(=O)=O)cc1 N1(C(=O)SCCNC(C)=O)CCC(CCCNC(=O)C=CCOC(C)(C)C)CC1 C1(C)(C(=O)NCCCCN(C(C(CC#C)C)=O)C)CCC12CCC2 c1(C(N2CCCC(CNC(C(C)(C)OC)=O)C2)=O)cc2c(C)ccc(C)c2[nH]1 N1(C(C(=O)NC(CC)CCO)C)CCN(c2ccccc2)C(C)C1 CC1COCCC1C(N1CC(CCNC(c2ccc(C(F)(F)F)o2)=O)C1)=O C(=O)(CCCCC(C)C)NC(c1cn(C)nn1)C(=O)N(CC)CC1CCOC1 C1(CC)C(NC(=O)Cc2cc[nH]n2)CCCN1C(=O)Cc1cnccn1 C1(NC(c2nnc(O)nc2O)=O)CC2CC1CC2C(=O)NC1C=CCCCC1 N1(C(CCc2ccn(C)c2)=O)CCC2CCN(C(=O)C=CCn3cncn3)CC12 c1(C(N(CC(=O)NCC2CCOCC2)CC)C2CC2)ccc(F)cc1 C1(CNc2cc(N(C)Cc3cc(-c4ccco4)on3)ncn2)COC2(CCC2)C1 N1(C(CC(C)(C)C)=O)C2CCC1(c1cn(CCOCC3CCCO3)nn1)CC2 N(C(=NCC(C)(C)CC)NCC1CCOC1)CC(C1CCOCC1)OC c1(CC)ccc(C(=O)NCCCN(CCO)C(c2cc(C)c(C)s2)=O)c(C)n1 Cc1ccnc(O)c1C(=O)NC1CCC(NC(C2CCC(C)(C)CO2)=O)CC1 CC1CC(CC(=O)NCCc2noc(=O)n2C)CN1C(c1cnc[nH]1)=O C1(CCC)CN(C(=O)CN(CC(C)C)C)CCN1C(=O)C(C)N(C)C(C)=O C#CC(C)(C)C(=O)NCc1cccc(C(=O)NCC2CC2Cl)n1 N1(C(c2c(C)sc(Br)n2)=O)CCCC(NC(=O)C=CC2CC2)C1C C1(C(=O)NC(C2CCCC2)CC)CC(NC(=O)Cc2ncccn2)C(O)C1 C=C=C(C)CC(=O)NCCCN(C(=O)CC1NC(=O)NC1=O)C(C)C CN(C)S(=O)(=O)N(C)CC(=O)NC1CC12CC(NC(=O)CC1CC(C)(C)CO1)C2 c1(C(N2CCC(NC(CC(COC)(C)O)=O)CC2C)=O)cc(Cl)cc(C)c1C CCC(CN(C)C)CC(=O)NCC1(CO)CCCN(C(=O)COCC2CC2)C1 Cc1ccc(C=CC(=O)NC(C)CC(C)NC(c2scnc2C(C)C)=O)o1 C(C(O)C(=O)NCCOCCC(=O)NC(C1CCCO1)CC)=CC O=CN1CCCC1C(=O)NC(c1cccnc1)C(=O)NCC=CCO C1(NC(CSCc2nc(C)sc2)=O)CCN(C(C2CCOC2=O)=O)C12CCC2 C1(CNC(COCC(=O)OC)=O)CN(C(=O)C(C)COC)CCC12CCC2 Cn1nnc2c1C(C(=O)N1CCCC3(NC(c4cnccn4)=O)CC3C1)CCC2 C1(NC(C2CC(=C)CN2Cc2ccc(N(C)C(C)C)cc2)=O)CCCCC1(F)F c1(C(=O)NCCN(C(=O)CC2C=CCC2)CCOC)nc(C(C)(C)C)cs1 N1(CC)CCOCC1C(=O)NCCCC(C)NC(c1cc(-c2ccoc2)[nH]n1)=O C1(C(=O)NC(c2cccnc2)CO)CC(O)CN1C(c1cccc(CO)n1)=O N1(C(C(C=CC)O)=O)CC2(CC(C(=O)NC(CC)(CC)C(N)=O)CO2)C1 C1(C(=O)NCC2(O)CC(CNC(CCC=CC(C)C)=O)C2)CC2CCC1O2 Cn1cc(CC(=O)NC2CCN(C(=O)CCn3cnnn3)C2)cn1 c1(C(N2CCC(O)(CNC(c3cc4n(n3)CCC4)=O)C2)=O)cncc2c[nH]nc12 c1(OC)nc(C)c(C(=O)NCC(CO)NC(=O)CCOC(C)C)s1.C12CC1C2 c1(C(N2C(C3CN(C(CCOC)=O)C3)CCCC2)=O)ncc(Cl)cc1F N1(C(CN2C(C)CCC2)=O)CCC(NC(C2(C)CCCN(C)C2)=O)CC(C)(C)C1 N1(C(c2cc3n(n2)CCC3)=O)C2CCC1C1CC1(NC(=O)C(F)(F)C(F)F)C2 c1(-c2ccc(C(=O)NCC3(NC(C(CC)N(C)C)=O)CCC3)o2)ccccc1Cl C(=O)(C(O)CNC(=O)C(C1(O)CCCC1)F)N(CCF)CC N1(C(C(CC=C)OC)=O)CCCC(O)(CNC(c2ccc3ncsc3c2)=O)CC1 C1(NC(C2Cc3cccnc3C2)=O)CN(C(C2CC3(CC3)C2)=O)CCC12CCC2 CC1(C(=O)NC2CCN(C(c3cccc(Cl)c3)=O)CC2C(N)=O)CCCCCC1 C1(C(=O)OC(C)(C)C)CC(S(C)(=O)=NC(=O)C2C3CC(=O)CC23)C1 C=CCCCC(C)(C)C(=O)NCC1CCN1C(c1cnc(C)[nH]c1=N)=O O=C1CCCC(C(=O)NC2CCN(CCNC(=O)CN3CCCCCC3)CC2)O1 N1(C(CCCCSC)=O)CC2CCC2(CN(CC(C)C)C(C2CCCCN2)=O)C1 c1(C(=O)NCC2CN(C(=O)Cc3cc[nH]n3)C3CC23)cc2c(Cl)cccc2s1 CC1CC(c2nnnn2CCCF)(NC2CC2)CN1Cc1occc1C1CC1 c1(-c2cc(C)c(CNC(=O)OC(C)(C)C)c(Cl)c2)cc2ncnn2cn1 CCC(C)(CC)C(=O)NC(C1CCCC1)CNC(=O)CCCN(C)C CC(C)(C)CC(O)C(=O)NCC1(F)CN(C(=O)COc2nc(O)nc(O)n2)C1 CC1CC(C(=O)NCCCN(C2CC(NC(C3(n4cccn4)CC3)=O)C2)C)=NO1 C1(N(C(C(C)(F)F)=O)C)CCC(NC(C2CCCCC2c2nc[nH]n2)=O)CC1 Cc1nccnc1C(N1CCCC1C1CCN(C(=O)CC2CCC(=O)N2C)C1)=O C1(C(N(C(C)C(=O)OC)CCC)=O)CN(C(c2cc(OC)no2)=O)CCC1O c1(SCCOC)ccccc1F.n12nnnc1C2(C)C.c1(CN)nncn1CC c1(C(=O)NC(C)CCN2CCOC2=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(C(COCC)C)=O)CCN(C(=O)Cc2c[nH]nc2O)C2CCCC12 N1(C(c2ccc(NC)cc2Cl)=O)CC(CNC(=O)CN2CCC2C)CC(C)(C)C1 c1(C(N2CC(CNC(C(C)C(F)F)=O)C(O)C2)=O)ccc2cc[nH]c2c1F C1(C)(C(=O)NCC(C(C)C)NC(C2CC(C3CC3)C2)=O)CCN(C)CC1 c1(C(N(CC(C)NC(C2CCC(=C)CC2)=O)CC)=O)cn(C)ccc1=O N1(C(C(CCOC)NC(c2ccc(C)s2)=O)=O)CC2(CC(NC(C)=O)C2)C1 C1(CCNC(CCSCC(C)C)=O)COCCN1C(C1(C2CCCCO2)CC1)=O c1(C(N(CCNC(C2CC3(CSC3)C2)=O)CC)=O)cn(C)c2ccc(F)cc12 c1(C(=O)OC)cccc(NC(=O)N2N3CC(C(C)C3)N2)n1.c1(SC)scnc1C c1(C(=O)NC2CC(NC(C(COC)CC(C)C)=O)C2)sc(S(C)(=O)=O)nc1C C1(NCc2cccc(C(=O)OCC)c2)CS(=O)(=O)CC1NC(c1ccccn1)=O c1(CC(=O)NCC2(C)CCN(C(CCC(CC)C)=O)CC2)cn2ccccc2n1 C1(NC(c2cnc3ccoc3c2)=O)CN(C(=O)C=CCO)C2(CCOCC2)C1 c1(C(=O)NCC(CNC(C(C2CCC2)OC)=O)CO)cccc(C(F)(F)F)c1O N(C(=S)NNC(=O)C1CCOCC1)C(C=C)C C(=O)(C1CCCc2c1ncn2C)N(C(C)C(=O)NC1CCN(C(C)=O)C1)CC C1(c2ccc(OC)cc2)(Cc2nnnn2Cc2ccccc2F)CC2(CCC2)C1 c1(C(=O)NC(CC)CNC(=O)CC2CCCO2)c(OC)ccc2cccnc12 c1(CC)ccc(C(=O)N(C(CNC(=O)C(C)(C)OCC(F)(F)F)C2CC2)C)s1 C1(C)(N(C(C(C2CCC(=O)N2)C)=O)C2CC2)CCCC1.C12CN(C1)C(=O)CO2 N1(C(c2cc(CC(C)C)n(C)n2)C(=O)NCC(F)F)CCN2CCC1CC2 Cc1cccc(CSCC(=O)NCC2CC(NC(=O)C3=COCC3)C2(C)C)c1 C1(NC(C(C)OCCC(C)C)=O)COCCN(C(C2CCCCCC2)=O)C1 N1(C(C)C)CCOC(C(=O)NC2(CNC(=O)C(C)C(C)O)CCCCC2)C1 C(=O)(C(C)(C)CS(N)(=O)=O)NCC1N(C(CCc2cc(C)[nH]n2)=O)CCN(C)C1 CN1CCOCC1CC(N1CC(O)(CCNC(c2cc(C(F)F)no2)=O)C1)=O c1(C(c2ccccc2NS(C)(=O)=O)NC(CN(C)C)=O)c[nH]c2ccccc12 c1(C(C)=O)ccc(C(=O)NCC2C=CCN2C(=O)COCC2CC2)cc1C C(=O)(C1CCc2c[nH]nc21)N1CCN(C(c2c(C)nn(CC)c2C)=O)CC1CF c1(C(=O)NCc2c(C(N3CC(C)S(=O)CC3)=O)con2)coc2ccccc12 C1(CC(=O)N(CCOC)C)CN(C(=O)C(C(C)C)Sc2ccccc2)CCO1 CC(C)C(O)C(C)C(=O)NCCCCCCC1CC1.C1C(O)C(=O)N1 c1(C(N2CCC(C)(O)C2)C(=O)NC(c2ccccc2)(COC)C)ccnc(Cl)c1 N1(C(c2cc(CNC(C3(C(=O)NC4CC4)CC3)=O)cs2)=O)CCC(CO)C1 C1(NC(=O)Cc2cnc[nH]2)CCN(C(c2ccc(O)nn2)=O)CCC1CO N1(C(C)=O)CC(CNC(c2ccc3nn[nH]c3c2)=O)OC2CCCC12 Cc1sc(C)c(C(=O)NCC2CCCC2NC(=O)C=CC2CC2)c1Br CC1(NC(=O)C(Cl)=CCl)CCN(C(=O)Cc2cccc(C(N)=O)c2)CC1 Cc1ccc(N)c(C(=O)NC2CC2NC(=O)CCC2CCCCC2)c1 C(=O)(C(C(C)NC(c1cncc(C#N)c1)=O)C(C)C)NCCC(C)C c1(C(=O)NC(C)CNC(C2CCCCC2C)=O)c(Cl)cc(Cl)c2ncccc12 CC1CN(C(c2cncc(N)c2)=O)CCCN1C(=O)CCC(C)(C)F c1(CNC(=O)N(Cc2cccnc2)CC2CC2)cc(C(C)(C)C)no1 Cn1nc([N+](=O)[O-])c(Cl)c1C(N1CCC(CCNC(C2(CC(F)F)CC2)=O)C1)=O c1(CCNC(CS(N)(=O)=O)=O)cc(O)nc(CNN2CCN(CC(F)F)CC2)n1 c1(C(N(C(C)CN(C(=O)CN(C2CCSC2)C)C)C)=O)ccc(CO)c(F)c1 c1(C(N2CC(C)CC(NC(C(CCSC)O)=O)C2)=O)cc2c(Cl)nccc2o1 c1(CNC(C2CCOC2OC)CC)ccc(OC)c(Br)c1 CC1CN(C(=O)C2=CCCN(C(=O)C3=C(Cl)CC3)C2)Cc2nncn21 c1(C(N2CC(NC(C(CC)(CC)OC)=O)C(OC)C2)=O)cc(N)c(F)cc1F c1(NC(C2CC3CC3N2C(=O)C=Cc2cnccn2)=O)ccnc(F)c1F N1(C(CC(C)SC)=O)CCCC2(CNC(c3cnc4c(c3)CCC4)=O)CCCC12 C1(C)(CC(NOCC(=C)Cl)=O)CCN(C(=O)C(CC)OCC)C1 c1(C(C2CC2)OC)nc(CCc2ccc(C)cc2)n(-c2nc(Br)nn2C)n1 N1(C(CC(CC)CC)=O)CCN(C(=O)CCCCCSC)CC(O)C1 C1(C(=O)NC(C2(OC)CCC2)C)CC2CCC(C1)N2C(C12CSCC1C2)=O C(=O)(C(C)C(O)C(C)C)N1CCC(NC(c2c(C)nncc2)=O)C1(C)C Cc1cccc(C(N2CCN(CC(N3CCOC(CCO)C3)=O)CC2)=O)c1I O=C1CCC(CNC(=O)COC2CN(C(=O)CCC3CCC3)C2)N1 C(=O)(C#CC1CCCCO1)NC1C(NC(=O)COc2ccc(Cl)cc2F)CCC1 c1(-c2ccc(OCOC)cc2)n[nH]c(=Nc2cccc(F)c2C(N)=O)o1 C1(C(=O)NCCCNC(Cn2cccc(C)c2=O)=O)CCC2CCC(=O)N12 c1(C(CNC(=O)CSS(C)(=O)=O)NC(C2CC(CC)C2)=O)cc(F)cc(Cl)c1 c1(C(=O)NC2CCN(C(C(CC#C)O)=O)CC(O)C2)cccc2c1OCC2(C)C c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C3CCC(=O)N3)C)C2)cc(Cl)n1 c1(OCC2CCCN(CCC(=O)Nc3ccccc3F)C2)cccc(F)c1 c1(OCC(=O)NCCCCCn2cc(CCCCO)nn2)ccc(Br)cc1Cl CCC(C)(C)C(C)CC(=O)NC1CN(C(C2(Cc3cnn[nH]3)CCC2)=O)CC1C c1(NC(C2C(C(=O)NCc3ccc(O)c(Cl)c3)C2)=O)ncc(O)cc1Cl n1(CC(C)NC(C2CCC2C(=O)O)=O)cc(-c2cnn(C3CCCC3)c2)nn1 c1(C(=O)NC(CC=C)CNC(C2CSC2)=O)cc(OC)ccc1C CC1CC(C(=O)NCc2ccnc(N3CCN(C(C4C(C)C4C)=O)CC3)c2)=NO1 c1(C(=O)NC2CC(C)N(C(=O)C=Cc3ncc[nH]3)CC2)ccc2ccccc2c1 Cc1ccc(CC(=O)NC2(CNC(C3CC(C)(F)C3)=O)CCOC2)cc1[N+](=O)[O-] N1(C(c2ccc(OC)cc2)CC)CCCC2CCN(Cc3nccn3C)CC12 C1(NC(C2(OC)CCSC2)=O)CCN(C(=O)C=Cc2ccncc2C)CC(O)C1 c1(OC)ncc(C(N2CCCC2CNC(=O)C(=Cc2cnc[nH]2)C)=O)cc1C C(=O)(CC(C)(C)C(F)F)NC1CCCN(C(C(Cc2ccccc2)OC)=O)CC1 Cc1ccc(C(=O)NCCCC(C)(C)NC(=O)Cn2cc(Cl)cn2)c([N+](=O)[O-])c1 CC(C)C(C)(O)C(=O)NCC1CCCN(C(C2C3CC4C(C3=O)C24)=O)CC1 c1(OCC(=O)NCC(CC)NC(c2cnc(NC(C)=O)nc2)=O)ccc(F)nc1 c1(OC)cnc(Cl)c(C(N2CC(F)(C(=O)Nc3ccc(C(C)=O)cc3Br)C2)=O)c1 C1(NC(CC(C)c2ccco2)=O)COCCC1NC(=O)CCc1nnc[nH]1 N1(CCNC(=O)C2=CCSC2)CCCN(C(=O)CC2NC(=O)NC2=O)CC1 C1(C)(CNC(c2ncn(CC)c2)=O)CCN(C(C2CCOCC2(C)C)=O)CC1 Cn1nc([N+](=O)[O-])cc1C(N1CCCC(F)(CNC(=O)CN2CCCC2=O)C1)=O C1(C)(C(=O)NC(C=CC(=O)NCC(CC)CC)C)CCC(C)CC1 C1(NC(C(C)C2CCCO2)=O)CN(C(C2CC23CCC3)=O)Cc2nccn2C1 C1(C2CC2)(NC(c2ccc(C)c(CO)c2)=O)CCN(C(c2cnco2)=O)C1 C(CCC(C)C(=O)NCC=CCNC(c1n[nH]c(C)c1O)=O)OC N1(C(C(C(CNC(c2ccc(C#C)nc2)=O)C)F)=O)Cc2ccccc2C1C C=CCCC(F)(F)C(=O)N1CCC(NC(=O)C(c2ccccc2Cl)(C)C)C1 N1(C(c2ccc(C)nn2)=O)CC2CCC(C1)N2C(c1cnc(C)s1)=O c1(OCCNC(C(C)OCC(=C)C)=O)ccccc1OC(F)(F)F C12(C(NOC(C(=O)OC)(C)C)=O)COCC1CN(C(C1CN(C)CCN1)=O)C2 C=Cc1cncc(C(=O)NCC(C)(O)CNC(=O)C(=Cc2ccco2)C)c1 N1(C(C2(CC#C)CC2)=O)CC(NC(c2cnn3cccnc23)=O)C(N=[N+]=[N-])C1 C=C=CCC(C(=O)N1CC2CC2(NC(C2CC(C)C2)=O)C1)NC(=O)OC(C)(C)C C(CNC(c1ccn(C2CCOCC2)n1)=O)(CC)(CC)NC(C1C(CC)C1)=O C(=O)(C1=CC2(CCOC2)C1)NC(CNC(C1=C(C)OCCS1)=O)CC(C)C C1(F)(CNC(CC2(COC)CC2)=O)CCN(C(=O)OC(C)(C)C)CC1 Cc1cc(=NCC(C)(C)CC2CC2)[nH]c(=NCC2CC3(CCCCCC3)CO2)[nH]1 n1(CCCC)cc(C(=O)NCC2CC(NC(=O)C(C)C3CCCO3)C2)nn1 CC1(C)CCN(C(c2cc(CNC(=O)C=CCN3CCCC3)on2)=O)CC1 N1CCC(Oc2cc(C3C(C(C)(C)C)CNC3)ncn2)CC1.c1(O)cccnc1 c1(OC)ccc(C(N2CCOCC2CNC(C2CC2C(F)F)=O)=O)c(Cl)n1 c1(C(=O)NCC(CC)NC(=O)CC2CSCCS2)cnc(C(N)=O)cn1 CC1CN(C(c2cn(C)nc2O)=O)CC(C)CN1C(c1ccnc(S)c1)=O Cc1nccc(CCC(=O)NCC(O)CN(C(=O)Cn2ccc(C(F)F)n2)C)n1 C1(C(C(=O)NCC=C)F)CCN(C(=O)C(c2ccccc2)O)C1 N1(C(c2scc(OC)c2)=O)CCN(C)CC1C(=O)N(C1CCOC(C)C1)C Cc1cc(C(=O)NC(C2(O)CN(C(c3cccnc3C)=O)C2)C)c(O)nc1C C1(C(=O)OCC)(C(N2CCC(CC3CC3)C2)=O)CCCCO1 N1(C(C2C(C)=CCS2)=O)CC(C(=O)NCCC2CCCN(C)C2)CCC1(C)C c1(CN(C(CC)C(=O)OC)C)ccc(S(=O)(=O)N(C)C)cc1 C1(C(C(=O)Nc2ccc(OC)cc2)N(CC(C)OC)CC)CS(=O)(=O)CCO1 c1(C(=O)NC2CC(NC(C(=O)NCC)=O)C2)ccc(S(=O)(=O)CC)cc1 n1(CC)ncc(Cl)c1C(=O)NC1(CNC(c2ccn(CC(F)(F)F)n2)=O)CCC1 N1(C(c2ccco2)=O)C2CCC(C1)N(C(C1CCCC(O)C1)=O)C2 C1(C(=O)NC2CC(OCC(=O)NC(CC)C(N)=O)C2)CCSC(C)C1 C1(C(NOCC(=O)OC)=O)CN(C(c2ccsc2Cl)=O)CC1C(C)C Cc1nn(C)cc1CC(=O)NC(C)CCC(=O)N(C)CC1CCCOC1 C(=O)(C1=CC2CC(C1)CC2O)NCC1(F)CC(CNC(c2ccc(C)o2)=O)C1 Cc1cn2nc(C(=O)NC3CN(C(=O)C(C)O)CC4(CCC4)C3)cc2c(=O)[nH]1 N1(C(c2c(C)nn(CC(F)F)c2)=O)CCN(C(=O)CO)C(c2cccnc2)C1 C(=O)(C1=CCCOCC1)N(C1CC1)CC1N(C(C2ON=C(C)C2)=O)CCC1 C1(NC(COCCC=C)=O)CCN(C(c2csc(Br)n2)=O)CC1C(C)C C(=O)(C#CC1(C)CCCO1)NCC1C(C)(C)N(C(C2C3CCC(=O)C23)=O)CC1 N#CC1CN(C(=O)COC2CCCC2)CCN1C(=O)CCn1cncn1 C(C(=O)N(CC)CC1(C)CCCC1NC(C1CSC1)=O)(C(C)C)OCC CCN=C(NCC1(S(=O)(=O)N(C(C)(C)C)C)CCC1)N1CCC(C(=O)OC)C1 N1(C(n2c(C(C)CC)nc3ccccc23)=O)CCOC2(CCS(=O)(=O)C2)C1 C1(C(N(C2CCCN(C(c3c(OCC)ccs3)=O)C2)C)=O)Cc2nccn2C1 N1(C(COCC(=O)NC)=O)CCC(O)(CCNC(c2cccc(F)c2C)=O)CC1 c1(C(=O)OCC)ccc(NC(=O)C(C)COC(C)(C)C)cc1Br N1(C(C2(OC)CC2)=O)CCC(O)(CCNC(c2nocc2Br)=O)C1 C12(C(N(c3ccccc3Oc3ccc(Br)cc3)C(C)C)=O)CCCC1C2Br CCCC(C)(O)CNC(C1(CC)CCN(C(=O)COC2CC2)C1)=O C1(NC(c2cnnc(Cl)c2)=O)COCCN(C(c2ccc(Cl)c(F)c2)=O)C1 c1(C(=O)NC(CCNC(COCC)=O)C(C)(C)C)cccc2c1CCCC2=O CC(CCCCNC(=O)C(C)(C)F)NC(=O)C(Oc1ccccc1)OC c1(CC)c(C(=O)NC(c2cn(CCC(C)C)nn2)C)nc2n1CCCC2 CC1(C(N2CCN(c3cc(C4CCC4)no3)CC2)=O)CCC(F)(F)C1.CC#N c1(C(N2CC(NC(CSCCN(C)C)=O)C(F)CC2)=O)ccc(F)c2ccsc12 Cc1cccc(CC(N2CCC(CN(C)C(c3ccns3)=O)C2)=O)c1 C(=O)(CC(C)C(C)C(C)C)N1CCC(=CCNC(C2(OC)CC2)=O)CC1 CCC(C)C(C(=O)NC1CCCC(NC(=O)C2=COCCO2)C1)SC N1(c2nnc(C(C)NC3CC3)s2)CC(C(=O)O)C(C)C1 N1(C(C)C)CCCC1C(=O)N(CC(C)NC(=O)C(F)OC(F)(F)F)C C1(NC(COCc2onc(C)n2)=O)CN(C(C2CC3(C2)CC3F)=O)C2(CCC2)C1 c1(C(N(C2CCN(c3cc(-c4ccccc4)ncn3)C2)CCC)=O)cc(Cl)cn1C c1(C(N2CCC(CN(C(C(C)OCC)=O)C)C2)=O)cc(Br)cnc1O C(=O)(C(F)(F)C1CCCC1)NCC(C)N(C)C(C1CC(OC(F)F)C1)=O C(=O)(CCC(C)NC(c1ncncc1Cl)=O)NCCCC(C)C N1(CCCNC(C2C(C(=O)NC3C(c4n(C)ncc4)C3)C2)=O)CCC(=O)NC1=O c1(C(N2CCC(N(C(C3CC(O)C3)=O)CC)C2)=O)cc(C)c(F)cc1F C(C(=O)N1CCC(C(=O)NC2CCCN(CCO)C2)O1)OCC=COC c1(C(=O)NCCC(C(C)C)NC(=O)C(=O)N(C)C)cc(F)c(Br)c(F)c1 Cc1cc(C(=O)NCc2cccc(OCC#N)c2)c(N)c(F)c1 C1(CC)CCN(C(c2cncc(O)c2)=O)C1C(=O)NOCC1CCCO1 C1(NC(C2(C)CC2(F)F)=O)CC2CCC1N(C(c1ccc(OCCF)cc1)=O)C2 CCC(O)C(C)C(=O)N1CCC(CC=C)(NC(c2ccc(CC(N)=O)cc2)=O)C1 CC1CCC(NC(c2cscc2C(F)(F)F)=O)CN1C(C1C(F)(F)C12CCC2)=O C1(CNC(C(C)=C2CCCC2)=O)(NC(=O)CCC2CC(C)(C)CO2)CCCCC1 Cc1cc(C(=O)NCCCC(O)C(=O)N(C)Cc2ccn(C)n2)ncc1N c1(NC(CN2CCC(C#CC)C2)=O)cc(O)c(C)cc1C C=CC(C)(C)C(=O)NC1CC(C)N(C(=O)C(c2cccc(C)c2)=O)C1 C1(CC(=O)NCC(O)CC2CCC2)CC2C=CC1C2.C12(CC)CN(C1)C2=O N1(C(=O)OC)CCC(CO)C1C(=O)NC(=O)CC1(F)CCC1.C1CN(C2CCC2)C1 Cn1c(C(N2CC(NC(=O)C=CC(C)(C)C)C3CCCC23)=O)cc2occc12 C1(NC(c2n(C=C)nnc2)=O)CCN(C(=O)C(=Cc2cccnc2)C)CC1F C1(NC(C=CC=CC)=O)CCCCC1NC(c1conc1C1CC1)=O c1(OC)ccnc(NC(C2CC2c2cn[nH]c2)=O)c1 c1(C(=O)NC(N(CCCN2CCCC2)C)=O)c(Cl)cccc1[N+](=O)[O-] c1(C(=O)NCC(CCNC(C(=O)NCC(F)F)=O)O)ccc2ccccc2c1F Cc1ccc(Cl)c(O)c1C(=O)NCC(O)CN(C(=O)CC=CC(C)(C)C)C N1(C(Cc2nc(C)sc2)=O)CC23CCCC2(C1)CN(C(c1cnco1)=O)C3 O=c1c2ccnn2cnn1CCc1ncc(CO)cc1Br N1(C(C2(COC)CCC2)=O)CCCCC(CNC(=O)CCCCCO)C1 c1(C(N(CCOCCCN(C(C(C)SC)=O)C)C)=O)cc2c(C)c(C)ccc2[nH]1 c1(C(=O)NC2C=CC(CNC(C(C)(C)CO)=O)C2)cnc2ccccn12 C(=O)(CC1=Cc2ccccc2C1)N1CCCC(N(C)C(C2(C)CC2(Cl)Cl)=O)C1 C=CCC(F)(F)C(=O)NC(C)CCN(C(=O)COc1ccc(C#N)cc1)C c1(NC(Cc2cccc(C(=O)OC)c2)C(=O)OC)nc(C)n2c1CCCC2 c1(C(N2CCN(C(C(C)=CC)=O)C(C3CC3)C2)=O)cnn2c1CC(C)CC2 N1(C(CCC2CC(C)C2)=O)CC2CC(C(=O)N(CCCO)CCCO)(C2)C1 c1(C(=O)NC2CN(C(C3CC(N(C)C)C3)=O)CC(O)C2)c(F)cc(F)c(F)c1F N1(C(CC(CC=C)NC(C2CCCC2OC)=O)=O)CC(C)(C2CCC2)C1 S(=O)(=O)(c1cccc(Cl)c1I)NC(c1noc(C(F)(F)F)n1)C C1(c2nc(COCC)nn2-c2nc(Br)nn2C)CCC2CC(C)CN2C1 C(=O)(CC(=O)NCC(O)CN(C)C(C1(CSC)CC1)=O)OCC c1(NC(CC2CC(=O)NC2)=O)nc2c(s1)CC(c1ccccc1)CC2 c1(C(N(C2CCN(C(C(c3cn(C)nc3)O)=O)C2)CCO)=O)ncc(Cl)cc1Cl C1(CNC(=O)CC2CC3(CC3)CO2)CC2CCC1N(C(=O)C=Cc1cc[nH]c1)C2 C1(CNC(C2CC(=C)C2)=O)CCC(C(=O)NC(c2ncc(C)o2)C)C1 c1(SC)ncc(C(N2CCC(O)(c3cccc(F)c3)C2)C(=O)NCCC#N)n1C c1(OC)ccc2nc(C(=O)NC3CN(C(C4(CO)COC4)=O)CC3F)ccc2c1 C1(C(=O)NC(C(C)NC(C(=O)Nc2ccc(C)s2)=O)(C)C)CC12CC(F)(F)C2 N1(C(C2(CC)CCCN2C(c2ncn(CC)n2)=O)=O)CCC2CCCC2CC1 C(CC(=O)NC(C(=O)NC(CO)C1(C)CC1)C1CCCC1)SC C1(NC(c2ccc(-c3cc(C)ncc3)cn2)=O)CCc2ccccc2C1 C(C(C(=O)N(CCCC(C)C)C)C(C)C)NC(c1cc(C(C)=O)on1)=O c1(C(=O)NC2(CCO)CN(C(C(CCC)OC)=O)C2)cnn(C)c1C#N N1(C(C2N3CC(C)N(CC3)C2)=O)CCC2(CC1)CN(C(=O)Cc1ncsc1Cl)C2 c1(C(N2CCC(F)(CNC(C3(O)CC3)=O)C2)=O)cc(Cl)cc2c1OCC2 C(c1ccc2c(c1)OCO2)=CC(=O)NCCC1(NC(C2CCSC2)=O)CCC1 N1(C(C(c2cc(C)cc(F)c2)C)=O)CC2(C)CN(C(=O)C(C)C(C)O)CC2(C)C1 CC1c2c[nH]nc2CCC1CNC(C12CC(c3ccccc3)(CO)C1C2)=O Cc1ccc(C(N)=O)cc1C(N1CCC(C)(NC(C2CC(C)(C)CN2C)=O)C1)=O c1(C(N2CCC(N(C(c3ccccc3)=O)CC)CC2)=O)ccc2oc(O)nc2n1 Cc1cncc(C(=O)NCC#CC(=O)NC2CCCCC2O)n1 C1(OCC)CN(C(=O)Cc2cccc(N)c2)CC1NC(=O)C(=O)NCCOC N1(C(C(CC)=CC)=O)CCN(C)C(C(=O)NCCN2CC3CCC2C3)C1 C(=O)(C1=CCCCC1)NCC(C1CCOC1)NC(=O)COC1CC(F)(F)C1 CC(C)(C)CC(C)(C)C(=O)N1CCOCC(NC(C2CCC=CCCC2)=O)C1 N1(C(C(C)C(C)O)=O)CCC(NC(=O)CNC(c2ccco2)=O)C(CO)C1 C(=O)(CC(C)(C)C(C)(F)F)NCCOC1CCN(C(C(C2CCOCC2)C)=O)C1 N1(C(C(CC)(C)C(=O)OC)=O)CC2CCN(C(=O)Cn3ncc(Cl)c3C)CC2C1 C1(C(N2CCCC(C(C)NC(=O)CCCC(C)=O)C2)=O)CCc2ccccc2C1 C(=O)(CCCCCC#N)N(CCC(=O)NCCC1(C)CCCC1)CCO C1(C(N(C(C)CNC(c2coc(Br)c2)=O)C)=O)CCCC(=O)N1 CC(C)(C)C(CNC(=O)CNC(N)=O)C(=O)Nn1cccn1 N(C(=NCCCS(C)(=O)=O)NCCS(=O)C(C)(C)C)C(C=C)COC C1(c2nc(SCc3ccn4ccsc43)nn2C2CCSC2)CCC2(CCOC2)O1 Cc1cc(C(=O)NC2C=CCN(C(c3ccc(O)nc3Cl)=O)C2)cc(=O)n1C C1(F)(C(=O)NCC(CCC)O)CCCN(C(c2cn(C)cc2C)=O)C1 C(=O)(CC(C)(C)CC(=O)N1CCN(C(c2n[nH]cc2Cl)=O)CC(C)(F)C1)OCC C1(C(N2CCC(NC(C(C)(C)n3ccc(C4CC4)n3)=O)C2)=O)CC(S(C)(=O)=O)C1 Cc1cc(Cl)ccc1OCC(=O)NC1CCCC1CNC(C1CC2(CCC2)C1)=O N1(C(COc2cc(C)on2)=O)CCCN(C(c2ccnc(C(N)=O)c2)=O)CCC1 C#Cc1cc(F)c(C(=O)NC(C)CNC(=O)C(O)C=C)cc1F C(=O)(C1=C(Cl)CC1)NC(C)CCCNC(c1ccsc1C(F)F)=O C1(NC(COC(CC)C)=O)CCN(C(=O)CCF)C1C C#CCC(C)(C)C(=O)NC1CCCC(CNC(=O)C(C)(O)CC)C1 C(=O)(C(C)(C)CN(C)C)NC1(C2N(C(c3nc(C(=O)OC)oc3)=O)CCC2)CC1 C1(CC(N2CC3C(C)C3C2)=O)CCCCC(=O)N1.C1(C(=O)NNC)CC2CC2C1 C1(NC(=O)CCC2CCN(C(=O)CC3CC3)C2)C=CCCC1CO C(c1cncnc1O)=CC(=O)NCC1N(C(C(COC)O)=O)CCOC1 CC(C)C(C(=O)NC1(CO)CN(C(c2cncc(C(F)F)c2)=O)C1)NS(C)(=O)=O Cc1nc(C(=O)NCC(C)CN(C(=O)C(C)C2CC2)C)cc(O)n1 N1(C(C(F)=CCC)=O)CCN(C(c2nc(C)ccc2F)=O)C(CCO)C1 CC1C(NC(=O)C(=O)NCC2CC2)CC2CCC1N2C(C1(O)CCSC1)=O C(=O)(C(O)CCNC(=O)C(CN(C)C)N(C)C)OC.C(=O)(C(CO)C1CC1)NC Cc1cc(C(=O)NC2CCC2C(N2CCC2(C)CN(C)C)=O)c(O)nn1 CC(C)CCC(CO)NC(=O)CN(C(=O)C(C)CC1CC1)C c1(OC)cc(C2(C(=O)NC3CC3CNC(=O)C3=C(C)OCC3)CCC2)ccc1C c1(C(=O)NCC(C)N(C(C(CC)F)=O)C)ccc2c(c1)C(=O)NCC(C)(C)O2 c1(OC)ccc(C(=O)NC2CC(C(=O)NC3(CO)CCC3)C2)c(Br)n1 C12(NC(CC(=C)C)=O)CC3CCC(C1C2)N3C(=O)CC(c1ccc(F)cc1)C C1(C(=O)NC2(C(=O)NC3(CC(N)=O)CC3)CC2)CC(CC2CC2)C1 C1(C)(CNC(c2scc(OC)c2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 C1(C(N(C2CCCN(c3cc(O)nc(O)n3)CC2)C)=O)CC2(C1)CC2(F)F C#CC1(O)CC(C(=O)N(C)CCN(C(=O)C[SH](CC(F)F)C(C)C)C(C)C)C1 N1(C(CCN(CC)CC)=O)CCC(C)(CC(=O)NC)C1.C1=CCNC1=O N1(C(C=C(C)Cl)=O)CCC2(CC1)CC2CNC(=O)C=CC1CCCN1C N1(C(C2N(C(=O)OC)C(C)C2)=O)CCCC(C(=O)Nc2cncnc2C(C)C)C1 C(=O)(C1CCCc2ccccc21)NCC(C)CNC(C1CC2C(C1)C2(C)C)=O Cc1ccnc(C(=O)NCCN(C2CCCC2)C(c2c(Cl)cnn2C)=O)c1N c1(C(=O)NCCOC2CCN(C(C(C)CO)=O)CC2)ccc(=O)n(C)n1 C1(C(C)NC(Cc2ccccc2)CC)(OC)CCNCC1 Cc1ccc(C(=O)NCC2CCCN(C(=O)Cc3ccnn3C)C2)c2c1CCC2 c1(OC)cc(CN2CCN(S(=O)(=O)c3cn[nH]c3)CC2)cc(C#N)n1 N1(C(CC(CC)(F)F)=O)CC(NC(=O)CCC#N)CC12CCCCC2 CCC(C)(CNC(=O)Cc1ncoc1C)C(=O)NCC(O)C(F)(F)F N1(C(C2CCN(C)CC2)=O)CC2(CC2)CC1C(=O)NC(c1ccc(Cl)cc1)CO C1(C(=O)NC2CC(=O)N(C)C2)(NC(CCCNC(=O)OC)=O)CCCC1C CC(C)(CC(F)F)C(=O)N1CC(CNC(C2CNC(=O)C2)=O)C(O)C1 CCCCC(O)C(=O)NCC1(COC)CCN(C(=O)CNC(N)=O)C1 N(C(O)=C1C2(C)CNCC(=O)N12)CC(C)(C)OC(C)C C1(NC(c2nc(OCC)oc2)=O)CC2CCC1CC2NC(c1cnnc(C)c1)=O c1(C(N2C3CC(NC(C(C)=C(C)C)=O)(C3)C2)=O)ccnc2ccc(O)cc12 N1(C(C(F)=C(C)C)=O)CCC(NC(=O)CC(C)(C)c2ccccc2)C(C)C1 C(=O)(CCS(C)(=O)=O)N(CC(C)N(C(=O)COc1cccnc1)C)C CCCC(CC)CCC(=O)NC(CNC(c1cnc2nc(C)oc2c1)=O)CC N1(C(C2(NC(c3cc(C)c(O)nc3)=O)CCOCC2)=O)CC(CO)CC(C)(C)C1 N1(C(C2(SC)CCC2)=O)CCOCC(F)(CNC(c2cn3c(n2)COCC3)=O)C1 N1(C(C(C)NC(=O)OC)=O)CC2CCC1C(CNC(=O)CC1COCCN1C)C2 N1(C(c2c(CNC(c3c(NC)ccnc3)=O)cc[nH]2)=O)CCn2c(C)cnc2C1 C1(CN(C)C(C2CC=CC2)=O)CCCN(C(=O)Cc2cn[nH]c2)C1 C1(NC(C(CC)NC(N)=O)=O)CC(CNC(C2(C(C)(F)F)CCC2)=O)CC1O C12(C(=O)NC(c3ccc(Cl)cc3)C)CCC(C(N3CCCC(O)C3)=O)(CC1)CC2 c1(C(N2CCC(NC(c3n(CC#C)ccc3)=O)(COC)C2)=O)nccc(Cl)c1F CN1CC2CCCC(C1)N2C(=O)C(C)(C)CCCNC(=O)CC1CCC(O)C1 N1(C(C(CSC)(C)NC(C2CCC3(CCC3)C2)=O)=O)CCC(O)C(C)(C)C1 O=C1CCC2(C(=O)NC3CC3CNC(C3C4CC5C(C4)C35)=O)SCCN12 c1(NC(C2(C)N(C(C(CC)O)=O)CCC2)=O)ncc(Cl)cc1[N+](=O)[O-] N1(C(C=C(CC)C)=O)CCC(CC)(NC(c2cc(OC)ccc2CC)=O)CC1 Cc1ccc(C(=O)NC2(CNC(c3cc4occc4n3C)=O)CC2)c(F)c1Cl C1(C(=O)NCC2(C)CCC(NC(=O)CCCn3ccnn3)C2)CN2CCN1CC2 C=C1CON(C(=O)c2ccc(SCCO)cc2)C1 C(=O)(C#CC(C)(C)CNC(=O)CC1COCCOC1)NC(c1ccnn1C)CC N1(C(c2cccc(C(C)C)c2F)=O)CC2(CCN(C(C3CC(N(C)C)C3)=O)CC2)C1 C(c1ccc(N(C)C)cc1)=CC(=O)N(C)CC1CN(C(C2(C)CCC(C)C2)=O)C1 C(C(C)N=c1cc(Cl)nc(-c2ccccn2)[nH]1)NC(CCc1c(C)cccn1)=O c1(CNC(C(CNC(=O)Cn2[nH]cnc2=N)OC)=O)cccc(C)c1F Cc1ccnc2nc(C(N3CCC(NC(C4CCS(=O)(=O)N4)=O)C3(C)C)=O)nn12 c1(C(=O)NC(C2(O)CCN(C(c3cc(C)no3)=O)C2)C)ncn2ccccc12 C1(CNC(C(C)CN2CCCCC2)=O)CCCN(C(=O)C(O)CN(C)C)C1 c1(OC)cnc(C(C)N)nc1.N1(C(C)=O)CCC(N2CCOCC2)CC1 c1(C(C)NC(C2C(NC(CC3CC(OC)C3)=O)CCC2)=O)ccccc1F C1(N(C(CC(CN(C)C)(C)C)=O)C)CCN(C(=O)C(C)(C)CO)CC12CC2 N1(C(c2nccnc2C)C(=O)NCC=C)CCC(N(C)C)C(C)C1 C1(c2nc(CC)on2)CCCN(C(=O)C=Cc2cc(OC)ns2)C1 c1(C(=O)NC2CN(C(C(C)NC(N)=O)=O)CC3C2C3)ccc2nc(O)oc2c1 Cc1cn2[nH]c(=NCC3CN(C(C4COC(C)(C)C4)=O)C3)sc2n1 N1(C(c2ncn(C)n2)=O)CCN(C(=O)CNC(=O)CCCCO)CC1CCO C1(O)(C(=O)NC2C(NC(=O)COC3CCOC3)CCCC2)CN2CCC1CC2 O(NC(=O)C1=CCC(NC(c2ccc(C#N)c(C)c2)=O)C1)CCCC C#CC1CCN(C(=O)C(C)CNC(=O)Cc2ccn(C)c2)CC1 c1(OCC)ccc(C)nc1C(=O)NCC1CN(C)CCN1C(=O)C(CC)SC c1(C(C)NCCOCC)cccc2c1OCO2 N1(c2nnc(COC)s2)CC2(CCC2)CC1CNC(C1CC2CCCC(C1)C2)=O C(=O)(C(C)(C)CC)NCC=CCNC(c1cn(CC(CC)O)nn1)=O N1(C(c2c(C)cccc2)=O)CCN(C(=O)Cc2ncn(C)c2C)C(C2CC2)C1 N1(C(c2c(CN(CCN(CCC)C)C)ccs2)=O)CC(OCC)CC(F)C1 c1(OC)ccc(C(N2CCC(C)C2CNC(=O)C(C)OCC(F)(F)F)=O)cc1Cl C12(C(N(C)Cc3cn(CCCc4ccccc4)nn3)=O)CC1CS(=O)(=O)C2 C1(C(=O)NCC(C)(CC(C)C)NC(c2c(C)cncc2)=O)Cc2ccccc2O1 N1(C(C#CC(C)C)=O)CCC(C(=O)NC(C)Cc2ccccn2)C(C)C1 C(CC(C(C)(C)C)N(C(C(C=C)CC)=O)C(C)C)NC(=O)COCCCCC CC1CN(C(=O)CCC(=O)c2cccc(Cl)c2)CCC1N(C(=O)CCC1CC1)C C1(C(=O)NCCOCC(C)C)(NC(C2CC(CC)C2)=O)CCN(C)C1 c1(CC)cc(C(N2CCCOCC2C)C(=O)NC2CCC2)ccc1Br c1(CCNC(NCCCC#C)=NC)ccccc1[N+](=O)[O-] c1(CNC(=O)C2=CCCC2)ccc2c(c1)CCC2NC(C1CC2CC2C1)=O C#CCCC(=O)NC(C)(CNC(c1coc(CO)c1)=O)CC c1(C(=O)NC2CCCN(C(C3(C)COC3)=O)C2)cc(=O)c2cc(F)ccc2[nH]1 c1(COC)ccc(C(=O)NCC2CC(O)(CNC(c3cnc[nH]3)=O)C2)o1 C1(CNC(C(F)=CCC)=O)CC(C)CCN1C(=O)C(CCSC)OC N1(C(COC(C)=O)=O)CCC2(CC1)CN(C(=O)CCc1c(C)n[nH]c1C)C2 N1(C(Cc2ccn(CC)n2)=O)CCCCC1CCN(C)C(c1nc(C)n(C)n1)=O C1(C(N2CC(C#N)C2)=O)COCC1NCCN(C(C(=O)N(C)C)=O)C(C)(C)C C1(NC(c2ccc(F)cc2Cl)=O)CCN(C(=O)Cn2cccc(O)c2=O)CC1F c1(C(=O)NCC2(O)CCN(C(C(CCC#C)O)=O)C2)ccc2c(c1)ncn2C c1(C(N2CCC(CN(C)C(c3sccc3Cl)=O)C2)=O)ncnc(O)c1F C=CCC(C)(C)C(=O)N1CC(C(=O)NCC2CC(=C)C2)CCC1C Nc1cccc(C(N2CCC(OCCNC(=O)CCN(C(=O)CO)CO)C2)=O)c1O c1(C(N(C)CC2CCN(C(CC=CC=C)=O)C2)=O)noc(C)c1I c1(SC)ccc(CCC(=O)NCCC2(O)CCN(C(C3(C)CC3(C)C)=O)C2)cc1 N1(C(c2noc(C)c2Br)=O)CCC(CNC(=O)C=CC2CC2)C(C)C1 C(=O)(C(F)CCC(C)C)N(C1CCN(C(C2(OC)CCOCC2)=O)C1)CC1CC1 N1(C(C=CCOC)=O)CCC2(CC1)CC(NC(=O)C(C)CC(C)(F)F)CO2 N1(CC(=O)NCC2C(C)CCCC2)CCC(C(F)(F)F)C(F)(F)C1 C1(CNC(c2c(CC)nn(C)c2)=O)CN(C(C2(C)CCC2)=O)CCC1C CCC(C(=O)NCCCCSC)(c1ccccc1)N(C)C C1(NC(c2c(C)[nH]nc2C(C)C)=O)CCCCN(C(C2CCSC2)=O)C1 c1(C(=O)NC(CNC(C2CCC(CC)CC2)=O)C)ccc2c(ccn2C)c1 c1(C(N2CCN(C(Cc3cnc(C)[nH]3)=O)CC2C(F)F)=O)ncc(C#N)cc1Cl C(=O)(C#CC1(C)CCCO1)NCCCN(C(c1c(OC)ccc(C(F)F)c1)=O)C C(CCCCOC)(C(=O)NC1CCOCC1)N(CC)Cc1cccc(Cl)c1F C(=O)(C1Cc2ccccc21)N1C(C(=O)NCC(C)(C)F)CCC1 C1(NC(CC(CNC(CC2N(C)CC=CC2)=O)C2CC2)=O)CCC2(CCCC2)C1 C1(C(=O)NCc2n(CC)cnc2)CCC2CCC1N2C(c1cnnn1C1CC1)=O C(=O)(CC(c1ccccc1)C1CC1)NC1CC(N(C)C(C2CC2(F)F)=O)C1 N1(C(C(CC(C)C)NC(C)=O)=O)CCCN(C(c2ccccn2)=O)C(CO)C1 c1(CC)n[nH]cc1C(=O)NCC(CC)NC(c1cnc(-c2ccccc2)o1)=O C1(O)(c2nc(CC)on2)CCN(Cc2ccc(C)nc2O)CC1 c1(CN(C(C2C3CCCCCC23)C(=O)NC(C)(C)C)C)cc(F)ccc1Br C1(CNC(C2CCC(CC)CC2)=O)CN(C(=O)CC2CCC(C)(C)O2)CC12CC2 c1(C(N2CCC(N(C(=O)CC3CCCCC3O)CC#C)C2)=O)cc(C)nc(O)c1 C(N=c1[nH]c(N2CCC(F)(F)C(F)C2)nc2c(F)cccc12)c1ccc(C)s1 Cc1nc(O)sc1C(=O)N(C(C)C(C)N)CCSc1ccccc1 C(=O)(C1=C(C)OCCS1)N1CCCC(C(N2CC(OC)C(O)C2)=O)C1C c1(C(=O)NC2CN(C(=O)CC3CCC3)CC2O)cccc([N+](=O)[O-])c1Br c1(C(=O)NC2(C(N3C(C)CSCC3)=O)CC2(C)C)ccc2c(c1)CC2 c1(OC)cc(NC(c2nc(-c3cccc(CC(=O)O)c3)sc2C)=O)ncc1OC CCCC(C(O)C(=O)NCC(CO)CC(C)C)NC(c1cnn(C)c1)=O C1(CNC(C2CCC(F)(F)C2)=O)CC2(CCC2)C1 c1(CC(=O)NCCCN(C(=O)CNc2ncccn2)C)ccc(F)cc1 c1(C(=O)NCCC(C)N(C(C(=O)Nc2ccc(C)cc2)=O)C)ncc(Cl)cc1F c1(C(CCC)NC(C2(N3CCOCC3)CC(O)C2)=O)cccc([N+](=O)[O-])c1 c1(C(C)=O)cccc(-c2cn(CC(=O)NCC(=O)NC3CCS(=O)(=O)C3)nn2)c1 c1(C(=O)NCCC(C)NC(=O)C(C)C2CC2)cccc2c1CCC2=O c1(OC)cccc2c(C(=O)NC3CCCN(C(=O)C(Br)=C(C)C)C3)csc12 CC1CCC(NC(C2CCC(F)(F)C2)=O)CN1C(=O)Cc1ccc(F)cc1 N1(C(C(c2cn(C)nc2)O)=O)CCN(C(=O)C=CCN2CCCCC2)CC1CO c1(C(=O)NCC(C2CC2)NC(c2cnc(C(C)OC)s2)=O)cccc2nncn12 c1(C(N(CC(CN(C(C(C=C)O)=O)C)O)C)=O)scc2c1CCCC2 c1(C(=O)NC(C(C)NC(=O)Cn2ncnn2)C)conc1C1(C)COC1 N1(C(C#CC(C)C)=O)CCC(CNC(C2(CC(C)=O)CCC2)=O)C(C)C1 C1(NC(CSCC(C)C)=O)CN(C(=O)CCc2cn(C)cn2)C2(CCCOC2)C1 C1(C)(C(=O)NCCCCCCNC(C2C(C)(C)C2)=O)CCCNS1(=O)=O C1(NC(COCCN(C)C)=O)CCC2CC1CN2C(=O)CC1CCCCC1(C)C C1(OC)(CNC(C2CCCN2C)=O)CN(C(c2scnc2CC(F)(F)F)=O)C1 Cn1nc2ccccc2c1C(N1CCCC(NC(=O)CCn2cnnn2)C1)=O C#Cc1cn(C)nc1C(=O)NCC1(O)CCN(C(=O)CC2CCCCC2C)CC1 C(=O)(CCC(C)N(C)C)NC(CC=C)CNC(C1CCOCC1)=O C12(CNC(C(C)(C)NC(C)=O)=O)CC3CC(CC(C3)C1NC(=O)C(C)C(C)C)C2 c1(C(=O)NC2(C(=O)NC3CC(COCC)C3)CCC2)cc[nH]c1C N1(C(C2CC(NC(c3c(C#C)cccc3)=O)C2)=O)CCc2cnccc2C1 C1(O)(CN(C(=O)CSC2CCCCO2)C)CCN(C(c2conc2C2CC2)=O)C1 C=CCC(C(=O)N1CC2CC1(CNC(C1COC(C)C1)=O)C2)c1ccccc1 C(C(CC(C)C)NC(c1ccc(C2(C)CC2)cc1)=O)NC(C1ON=C(C)C1)=O c1(C(=O)OC)ccccc1CN1CCOC(C)C1.C12CCCC1C(=O)N2 c1(C(=O)NC(C(=O)NC2CC3CC3C2)c2ccoc2)ccc(CO)nc1 Nc1ccc(C(=O)NC2CC(NC(=O)COC3CC3)C2)c(Cl)c1 c1(CC(=O)NCC2N(C(CSCC(N)=O)=O)CC3CC32)cccc2nsnc12 C1(C(=O)NC(C(=O)NC2C(C)(C)C2(C)C)c2ccco2)CC2(CCO1)CC2 c1(C(=O)NCC(CNC(=O)CC2CCOCC2)F)cnnc(-c2ccncc2)c1 CC1=NOC(CC(=O)NC2CC2NC(C2CC(O)C2)=O)C1 c1(C(=O)NC2(C)CCN(C(c3c(COC)cc[nH]3)=O)C2)cccc2nn[nH]c12 C#CC1CCCN(C(=NCc2ccc(OCC)nc2C)NCc2ccccc2)C1 c1(-c2ccc(C)cc2)n[nH]c(=NC2Cc3cccnc3NC2=O)s1 CCC(CCC(=O)NCC=CCC(N1CCOC(C#N)C1)=O)SC C(=O)(C1=NOC(CNC2(C3CCOCC3)CC2)C1)OC(c1ccc2c(c1)OCO2)C Cc1cc(N2CCCC(NC(c3cnn(CC(F)F)c3C)=O)C2C)ncc1C#N C1(NC(C2CCC(CNC(C(COC)(C)C)=O)CC2)=O)CCOC(C)(CC)C1 C1(NC(C(N2CCCCCC2)C)=O)(CNC(C2CCOC2=O)=O)CCCCC1 c1(NC(C23CC2CN(S(=O)(=O)Cc2ccc(Cl)cc2)C3)=O)ccc(CO)c(Cl)c1 N1(C(c2c(COC)nn[nH]2)=O)CCCC2(C1)CN(C(=O)CC13CCCC1C3)C2 C1(C(C)C(=O)N2CC(CCO)C2)CCN(C(=O)CN(C)C2CC2)C1 C1(NC(C(C)SC)=O)CN(C(=O)C=Cc2cncnc2O)CCC1O CCCC(O)CC(=O)NCCC1CCCN(c2ncn(C)c(=O)c2Br)CC1 CCCC(C)(C)CC(=O)N(CCCCCC(=O)NC(c1ccon1)(C)C)C C1(C(N2CCC(=CCNC(C3N(C)C(=O)CC3)=O)CC2)=O)CCCCCC1C(N)=O N1(C(C)=O)CC2(C1)CN(C(C13CC4CC1C3C4)=O)C2.C1CC(C#N)C1 [N-]=[N+]=NC1CC=CCC1NC(=O)CN1CCCOC(C(=O)O)C1 C(N=c1cccc(S(=O)(=O)NCC(C)C(C)C)[nH]1)C1(OC)CCOCC1 C1(C(=O)NCCNC(=O)NCc2cnco2)CS(=O)(=O)CC1c1ccccc1 C(=O)(CCCC(C)(C)CC)NC1C2CC(NC(C3(OCC)CCC3)=O)C(CC2)C1 N1(C(C)C)C2CCC1CC(C(N1CC(CNC(=O)C3=CS(=O)CCC3)C1)=O)C2 N1(C(C(C(C)C)SC)=O)CC(C)N(C(c2cc(C)c(C)cn2)=O)CC1C c1(C(=O)NCCN(C(C(CC)N(C)C)=O)C2CC2)cnc(OCCOCC)nc1 Cc1cc(C)[nH]c(=NCc2c(C3CC3)cnn2C)n1 C(=O)(C1=CCC(C)CC1)NC(C(=O)Nc1cn(CC(C)C)nc1)C1CCCC1 C#CC1CCCN(CC(=O)N(C2CCCCCC2)C(c2ccc(C)o2)=O)C1 C1(C(=O)NC2C(CNC(CCOCCC)=O)COC2)COc2cc(Cl)ccc2C1 Cc1ccc(F)c(C(=O)NC2CN(C(c3coc(Br)n3)=O)C(C)(C)C2)c1 CC(C)S(=O)(=O)C(C)C(=O)N(CC(O)CNC(=O)C=CCn1cncn1)C N1(C(C(=O)NC2CCOC2)C2(C)CC2)CCC(C)C(CC(N)=O)C1 C(COCc1ccccc1)(C(C)(C)C)NCC1CC(C)(COC)C1.c1(O)ccccc1Cl c1(C2CN2)cccc(Cl)c1.CON(C)CCNC1(c2cccnc2)CC1(C)C c1(C(=O)NC2CN(C(=O)C=C3CC3)CC23CC3)ccc2nc3n(c2c1)CCC3 n1(CC(=O)N(C)CC2CN(C(c3cccc(Cl)c3F)=O)C2)nc2c(n1)CCCC2 c1(N2C3CS(=O)(=O)C(C3)C2)nc2c(c(=NCC(Cl)=CCl)[nH]1)SCC2 N1(C(CC2CCN(C)C2)=O)CCOC2(CCN(C(=O)Cc3cnc[nH]3)CC2)C1 C1(NC(Cc2c(C)ncs2)=O)COC2(CCN(C(C3CCS(=O)(=O)N3)=O)CC2)C1 c1(SC)cccc(-n2nc(-c3ccccc3Cl)nc2C23COCC2C3)c1 C#Cc1ccc(C(=O)NCCCS(C)=O)cn1.C1CC(=O)NC12CCC2 C(CCCC(=O)N1CC(OC2CCN(C(=O)C(C)OCC)CC2)C1)OCC C1(CN2CCN(CC(=O)Nc3c(COC)cccc3)CC2)CC2CC1CC2O C(=O)(C(CNC(c1ccc(OC)nc1)=O)CC=C)NC(C=C)C(C)OC N#Cc1ccsc1C(N1CC(O)CC1CNC(=O)C(F)(F)c1cnc(Cl)s1)=O C1(N(C(C2(OC)CN(C(=O)Cc3ccc(OC)s3)C2)=O)CC)CCCN1C(C)=O CC(C)(C)CCCC(C(=O)NC1CCC1)N1CCOC(C2CCC2)C1 C12(NC(CN3C(C)CCC3)=O)CCCC1CN(C(=O)C=Cc1ccsc1)C2 C1(C(=O)NCC2(CNC(=O)C(F)CC3CCOC3)CCC2)CCCC12CCC2 S(=O)(=O)(c1cc(NC(=O)N(C)C)c(Br)cc1F)NC1CCN(N(C)C)CC1 N1(C(c2c(C)n(C3CCC3)nc2)=O)CC(C2(NC(=O)Cc3nccn3C)CC2)C1 C(=O)(CCCCN=[N+]=[N-])NCC1C(C)(C)C1CNC(=O)CC1(O)CCCOC1 CC(C)CCCCCC(=O)NC1CC12CC(NC(=O)CC13COCC(C1)C3)C2 C12(C(=O)NCCC(C)(C)NC(c3n(C=C)ncc3)=O)CCCC(=O)N1CCC2 CCCCC(C)C(=O)NCCC1CN(C(C2CC=CC(O)C2)=O)CCCO1 C1(CNC(CCN(C(C2(COC)CC=CC2)=O)CCO)=O)OCCCC1(C)C c1(C(=O)NCCC2(C(C)C)N=N2)nc(C(F)(F)F)oc1Br N1(C(C(CC)F)=O)CC2(CCN(C(C3CCSC3)=O)C2)C1 CC1=C(C(=O)NC(CNC(=O)C(=O)NCCSC(C)C)CO)CCC1 CC(C)C(O)C(=O)NCC(CC(=O)NCC1(C(N)=O)CCC1)C1CCC1 C1(C(=O)NCC(N2CCOCC2)C)CC(F)(F)CN1C(c1ncccn1)=O c1(OC)ccc(NC(c2ccc(C(=O)NC3CC(C)C3)[nH]2)=O)cc1C#N N1(C(CCC=CCC=C)=O)CCOC2CN(C(c3cnc4n3CCCC4)=O)CC12 C1(CCC(N2CC(OC(=O)NCC)C2)=O)C=CCN(C(c2ccn(C)n2)=O)C1 N1(C(CCSCC)=O)CCCCC1C(=O)N(C1CCOCC1C)C C(=O)(CCC(=O)NC1CN(C(=O)CSC(F)F)C1)Nc1nnc(CC)s1 Cc1occ(C(F)(F)F)c1C(N1CCCC(N(C)CCc2cccc(N)c2)C1)=O CCCCC(CC)C(=O)N1CCC(CN(C)C(C2C3CCCC23)=O)CC1 c1(CCC(=O)N(C)CC=CC(=O)O)cccc(NC(=O)N(C)C)n1.c1(OCO)ccoc1 C(=O)(CCCC(c1nnnn1C)NCc1cccc(OCC(N)=O)c1)OC C(=O)(NNC(=O)NC1CCCOC1C1CCNCC1)NC C1(NC(COCC(C)C)=O)C2CC1N(C(=O)CCc1ccc(Cl)s1)C2C C(=O)(CCC1CCc2ccccc21)NC1C(C)CN(c2nc(Cl)ncc2Cl)C1 c1(C(N(CCCN(C(C(C(=O)OC)C)=O)C)C)=O)cc2c(o1)CCCC2 C1(CC=C)(NC(c2cc(F)cs2)=O)CCCN(C(=O)CC2C=CCC2)C1 c1(C(N(CC(CNC(c2ccc(NC)cc2)=O)(C)C)C)=O)n[nH]c2c1CCC2 N1(C(c2c(C)nn(C(C)C)c2C)=O)C2CCC1CN(C(c1ccn(C)c1C)=O)C2 C(=O)(C1CCc2ccccc21)N1C(CNC(C2(COC)CCC2)=O)CC(OC)C1 N1(CCC)C(=O)NC(c2cc(F)ccc2C2CC2)C2=C1CN(n1cccn1)C2=O N1(C(C(C)C(C)O)=O)CCN(C(c2ccc(C(F)F)cc2F)=O)C(C(F)F)C1 Cc1nc2cc(C(=O)NCC3CC(F)(CNC(=O)CC4(C#N)CC4)C3)ccc2s1 c1(CC)nc(C)c(C(=O)NC2(CNC(=O)C(C#N)OC)CCCC2)s1 c1(C(=O)NCC(C)CN(C)C(C2(CCN(C)C)CC2)=O)ccc(Cl)s1 c1(NC(N2C3CCC2CC2(CC2)C3)=O)ccnc2c1CCCC2O Cc1cc(O)ncc1C(=O)NC12COC(CNC(C34CCC3C4)=O)(C1)C2 C(=O)(CC(C(F)F)N(C)N1CC(SC)C(C)(C)C1)OCC c1(NC(C2CC2CNCc2cc(C(F)(F)F)cc(F)c2)=O)cc(Cl)cc(Cl)c1F C(=O)(C(F)(F)CCn1cccn1)N1CCCC(C(N2CCN(C)CC2CO)=O)C1 C1(NC(COC)=O)CCCC(CNC(c2cn(C3CN(C)C3)nn2)=O)C1 c1(C(=O)NC(CN(C(C2(CC=C)CCCC2)=O)C)C)ccc(-c2cscn2)cc1 N#Cc1cc(S(=O)(=O)NCC(=O)Nc2ccc(-c3cc[nH]n3)s2)ccc1Br Cc1cc(OCC(C)C(F)F)cc(C)c1OC1CCOCC1 c1(C(=O)NCCCC(C)NC(C2CCCN2N=O)=O)noc2ncccc12 c1(C(=O)Nc2cccc(NC(c3c(C)occ3)=O)c2)c[nH]c(=N)nc1C C1(C(=O)NC2(C(N3CC(C(CC)C)C3)=O)CCCCC2)CC(=O)NC(=O)N1 C1(F)(CNC(C2C(C)C2)=O)CC(CNC(=O)Cc2csc(-c3ccccn3)n2)C1 Cc1noc(C)c1C(C)C(=O)NCC(C)CN(C)C(C1CC(F)C1)=O N1(C(c2nn(CC)c(O)c2)=O)CC(NC(c2cc(O)nc(O)n2)=O)CC2(CC2)C1 Cc1cccc(F)c1C(=O)NCC1(F)CC(CNC(c2cn(CCO)nn2)=O)C1 C1(O)(CN(C)C)CCN(C(C2CC(O)CN2C(=O)C=Cc2cn(C)cn2)=O)C1 C=CCCCC(C1CC1)NC(C1(NC(c2[nH]nnc2C)=O)CC(C)(C)C1)=O C1(C)(C(=O)NCC(C)CNC(=O)CC2(C(C)(C)C)OCCO2)CNC(=O)C1 N1(CC(C)C)CCCCC1CC(N)C(F)(F)F FC(F)(CCCn1nnnc1C(C1CC2CC2C1)NCc1nc(Cl)cs1)C(F)F N1(C(c2cnc(C(C)=O)s2)=O)CCC2CCC(C1)N2C(C1CCC1C)=O O=C(C#CC1CC1)NCCN(C(C1CC1c1occc1Br)=O)C1CC1 C1(CNC(Cn2c(C)cnc2)=O)CCN(C(=O)C(CO)N(C)C)CC1O c1(C(C2CC2(c2ccccc2)C(F)(F)F)=O)ncnc2[nH]c(Br)nc12 c1(C(=O)NCCC2CCCN(C(CCC(C)O)=O)C2)cccc(C#N)c1 C(=O)(C(C)CC(C)(F)F)N(C1CCCN(C(C2(OC)CC2)=O)C1)CC C1(C)(C(N2CCCC(NC(c3cnc(CC)s3)=O)C2)=O)CCCC1(F)F N1(C(C2CCCO2)=O)C2CCC1CC(CC(C)OC)C2.c12ccc(cc1)n2CC N1(C(c2c(C)nn(CC(F)F)c2)=O)CCC2(CCC2)C(NC(C2CCCC2)=O)C1 N1(C(c2c(Br)ccc(C#N)c2)=O)CCC2(CC1)CC(NC(C1(CCO)CC1)=O)C2 O=S(=O)(c1ccc(=NCC2CC3C=CC2CC3)[nH]c1)NC1CCC(F)(F)C1 C(=O)(C(O)CN1CCCC1)NCCC1(NC(=O)CSC2CCOCC2)CC1 Cc1cn2c(n1)CCC(C(=O)NC1CC(CNC(C3CC4(CCC4O)C3)=O)C1)C2 C1(C(N(CCCN(C)C)CCC)=O)CCCCC1CNC(=O)Cc1ccc(F)nc1 C1(C)CCCN1C(=O)C(Br)=C(C)C.C1(C(=O)OCC)(C(=O)NCCC2CC2)CCO1 c1(C(N(CCNC(=O)C(C)Cc2ccccc2F)CC)=O)c(C)cccc1F Cc1ccc2c(=NC3CCC3C)[nH]c(=NCCOCCc3ccccc3Cl)[nH]c2c1 c1(C(N(CCN2CCN(C(c3ccc(C)o3)=O)CC2)C)=O)cc(F)c(F)cc1F CC12CC(C1)C(C(N1CCCC(n3cc(CO)nn3)C1)=O)CO2 N1(C(c2c(C)coc2)=O)CCC(NC(c2cc(Cl)cc(C)c2N)=O)C(F)(F)CC1 c1(OCC)ccc(C)nc1C(=O)N(CCCOCCNC(=O)C=C(CC)CC)C CC(C)(CNC(=O)C(c1cccnc1)NC(=O)CCC1CCC(=O)C1)C(F)(F)F C1(CCNC(c2ccc(Cl)cn2)CC)CCC(C)(C)O1 Cc1cc(N)ccc1C(=O)NC1CCCCC1NC(C1CC1c1ccnn1C)=O c1(CN2C(C(=O)Nc3cc(C)no3)CCCC2)c(Br)ccc2c1OCO2 c1(CC)cccc(CNC(=O)NC2(C)CN(C(=O)CC3CSC3)C2)c1 N#Cc1ccc(=NCC2(F)CCN(C(C3CCOC3)=O)CC2)[nH]c1 c1(CNC2C3CC(C(=O)O)C(C3)C2)ccc2cccnc2c1 N1(C(C(c2cccc(Br)c2)C)=O)CCCC(C)(CNC(=O)C(C)(C)O)C1 N1(C(C(C)NC(N)=O)=O)CCC(CNC(=O)C(C)(C)CCCF)C(C2CC2)C1 Cc1cc(C)c(NC(=O)C(N2CCCC(C)(CO)C2)c2nc(Br)cs2)c(C)c1 c12ccc(nc1)C(=O)N1C(C(=O)OCCC(C)(C)C)CCC21.CCCN(C)C(C)C c1(C(=O)NCC(C(C)C)OCC)cc([N+](=O)[O-])cc(C)c1F C1(NC(CNC(CC(C)C)=O)=O)CCN(C(c2ccc(CN(C)C)[nH]2)=O)C12CC2 C1(CCC)CN(C(c2cccnc2)=O)CCN1C(=O)NC1CCC(C)CC1 c1(C(=O)NCCC2CCCN(c3nc(C)cc(OC)n3)C2)ccc(O)c(F)c1F c1(C2(C)CC2)cc(C(=O)NCCC2CSCCN2C(=O)C(C)(F)F)n(C)n1 N1(C(C2(C=C)CC2)=O)CCC(NC(=O)Cc2cc(F)cc(Cl)c2)C(O)C1 N1(C(CC2CC(C)(C)OC2)=O)CC(NC(=O)CCn2cc(Cl)cn2)CC(O)C1 c1(OC)ncnc(C(N2C(C(=O)O)(C(=O)O)CSC2c2ccccc2)=O)c1F c1(CC)cc(C(=O)N(C2CC(NC(c3cc(O)nn3C)=O)C2)C)cc(F)c1 Cc1nc2ccc(NC(=O)C(N3CCCC(NS(=O)(=O)C(C)(C)C)C3)C)cc2[nH]1 C(CC(=O)N1CCCOC(C)C1)(C(F)(F)F)NC(C1(CSC)CC1)=O N#Cc1cccc(C(N2CCCC2CCNC(c2cnn(C(F)(F)F)c2)=O)=O)c1 c1(C(=O)NCC(=O)NCCC2CC2)cccc2cncn12.N12CCN(CC1)CC2 C1(C(=O)OC)C=CCN(C(C(=O)NC2CCCCCC2)C2CCOC2)C1 c1(C(N2CC(N(C)Cc3ccc(C)cc3Cl)C2)=O)ccc(C#N)c(F)c1F Cc1cc(C(=O)NC2CCN(C(=O)CCC3CCOC3)C2C2CC2)cc(C)n1 CC(C)CC(CNC(C1(C)CC1)=O)NC(=O)CCCc1cccc(C(F)(F)F)c1 c1(C(=O)NCC2(OC)CN(C(=O)CCc3ccoc3)C2)cnc(C)cc1C C(=O)(C(O)C(F)(F)F)N(C1CCCN(C(=O)Cc2ccc(Cl)cc2Cl)C1)C c1(OC)cc(N)c(C(N2CC=C(CCNC(C3CSC3)=O)CC2)=O)cc1F C(C(CNC(c1cc(CC(C)C)[nH]n1)=O)CO)NC(C1CC(C)C1)=O c1(C(=O)NC(CC)C)c[nH]nc1CNC(=O)C(C)(C)OC c1(C(=O)NC2CC(C(=O)NCC3C(OCC)CC3)C2(C)C)cccc(O)c1F CCC(C#N)C(=O)N1CC(C)(NC(C2(CC(=O)OC(C)(C)C)CCOCC2)=O)C1 c1(C(=O)NC(C)CN(C)C(c2sc(C#N)cc2Cl)=O)cn2ncccc2n1 c1(CC(=O)NC2CC(OC)CN(C(=O)CCF)C2)ccc2c(c1)OC(F)(F)O2 c1(CC(N2CC3(CC(C(=O)NC4CCCCC4)C3)C2)=O)c(F)cc(F)cc1F N1(C(C(C(C)C)OC)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)CC(C)(C)C1 C1(C(=O)NC(c2nc(-c3ccsc3)no2)C)CCC(Cn2ccnc2)C1 Nc1cccc2cc(S(=O)(=O)NC3CCCC3)ccc12 Cn1c(C(N2CC3CN(C(=O)CCCc4cnn[nH]4)CC3C2)=O)cc2sccc12 N1(C(C2(CC#C)CCCOC2)=O)CCC(O)(CCNC(=O)CCC(C)SC)CC1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)C(NC(=O)Cc2cn3ccsc3n2)C1 c1(OCC)nn(C)cc1NC(=O)C#CCNC(=O)CC1CCC(C)C1 CCC(C(=O)NC(CNC(C1(F)CC1)=O)CC(F)(F)F)C(C)(F)F Cc1onc(-c2ccc(NC(c3cccnc3C3CC3)=O)cc2)c1C#N Cc1nc(O)[nH]c1C(=O)NCCC(C)NC(C1(F)CCCOC1)=O N1(C(C2N(C(C=Cc3cncc(C)c3)=O)CC2)=O)CCC(O)CC(C)(C)C1 C1(C(=O)NCC2(C)CCN(C(c3ncccc3F)=O)CC2)CC2CCC(C1)C2O N1(C(CC2C(NC(Cc3ccc(C)cn3)=O)CCC2)=O)Cc2ccc(C)cc2C1 c1(C(=O)NC2CCN(C(c3nn(C)c(CO)c3)=O)CC2F)ccn2nccc2c1 C(=O)(C1CCCc2cccnc21)NCC(C)CNc1nc(-c2ccccc2)ns1 CCC(C)C(O)C(C)C(=O)N1CCCC(CC)C1C(N1CCCC1CNC(C)=O)=O c1(C(N(C)CC2CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)cc2ccc(F)cc2[nH]1 C(=O)(C1OC(C)Cc2ccccc21)N(CC)CC.c12cccc(c1)NC2=O N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCN(C(=O)CCCN=[N+]=[N-])C2COCC12 c1(C(=O)NCC(CN(CC(C)C)CC)(C)C)cc(C)c(Cl)c(C)c1 c1(NC(C)=O)cnc(O)c(C(=O)NCC2CCC(NC(c3cc(C)on3)=O)C2)c1 N1(CC(=O)NC(C)CNC(c2cocn2)=O)CCOCC1=O N1(C(C=C(C)C2CC2)=O)CCCC2(CC(NC(c3sccc3CO)=O)CO2)C1 N1(C(CCC(C)OC)=O)CCCCC(NC(c2c(C(F)(F)F)coc2C)=O)C1 CCCC(C)(C)CC(=O)N1CC(F)(CNC(c2cc(S(C)(=O)=O)cs2)=O)C1 N1(C(=O)OC(C)(C)C)CC2(CCCC2CC(=O)Nc2ccccc2C#CC)C1 c1(OC)cccc2c1OCC2NC(=O)Nc1ccc(S(C)=O)cc1 N1(C(C=Cc2c(C)ncs2)=O)CCN(C(=O)COc2cccnc2)CC1C(C)C N#Cc1ccccc1C1CC1C(=O)NCC1(O)CCCN(C(=O)C=CCO)C1 CC(C)(CNC1CCC(NC(=O)CCCn2cc(CO)nn2)C1)C1=CCOCC1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC2CCN(C(=O)Cc3cncnc3)C2C1 CCC(CC(=O)NC1CC(C(=O)NC(CO)CC(F)(F)F)C1)C(F)F C(=O)(C(C)(O)C(F)(F)F)C(=O)C(O)CN1CCCC1.n12cc(nn1)C(=O)NC(C)C2 N1(C(C(CC=C)C)=O)CCCC(C)(C)C1C(=O)NC1=CC=C(N=[N+]=[N-])CC1 c1(N2CCCCC(SC)C2)nc(N2CCC(n3cc(C)cn3)C2)nc2c1CSC2 CCC(C)(O)C(=O)N(CCC(C)(C)NC(=O)Cc1ccc(C)o1)C N1(C(C=C(CCC)CCC)=O)C2CCC1CN(C(C1CC13CCC3)=O)C2 C(=O)(C1=CCCCC1)NC(C1CCCCN1C(c1cnc(C(N)=O)cn1)=O)C n1(C(F)(F)F)cncc1NC(=O)NCCOc1ccccn1.C1(N)CC1CO C1(NC(C=Cc2ccc(CC)o2)=O)CCN(C(=O)CCCC2(C)N=N2)CC(O)C1 CC1(C(=O)NC2CCCC2NC(c2ncc(F)cn2)=O)CCCCCC1 C1(OC)C(c2nnnn2Cc2ccco2)(Nc2ccc(F)nc2C)CC12CCC2 c1(CC)ccc2c(c1)NC2=O.c1(CS)cccc(O)c1Br.c1(SC)ccccc1F C#CCCC(=O)NC(C)CNC(c1nnn(-c2ccccc2)n1)=O c1(C(N(CCN(C(C2CC(CC)C2)=O)C)C)=O)cc(O)cc(F)c1F C12(C(=O)OC)CCCC1(C(N1CC(C)(NC(=O)CC3CC3(Cl)Cl)C1)=O)C2 C1(NC(C(C2CC2)NC(C(C2CCC2)OC)=O)=O)CCc2c[nH]nc2C1 c1(CC(=O)NCCN(C(c2cccc(OCCC)c2)=O)C)c(C)nc(O)nc1O C(CC(=O)N1CCC(NC(=O)CC(C)C(C)(C)C)C1(C)C)(C(F)(F)F)OC C1(N(C)C)COCC1NC(C1CCCN1C(N)=O)=O.C12CC(O)C1CC(=O)N2 c1(C(N(C(CCNC(c2c(C)cncc2)=O)C)C)=O)ncc(N)cc1Cl c1(C(=O)NC(C)CCN(C(=O)C(C)(Cl)Cl)C)cc2ccncc2s1 c1(C(=O)NCC(CNC(c2[nH]ccc2C)=O)OC)ncc2c(F)cccn12 c1(C(=O)NC2CN(C(C=C(CCN(C)C)Cl)=O)CC(O)C2)[nH]nc2ncccc12 C(=O)(C1=Cc2ccccc2OC1)N1CCC2(NC(CN(C)S(N)(=O)=O)=O)C(C1)C2 C#CCCC(O)C(=O)N(C1CN(C(c2ncncc2Cl)=O)CC1O)C C=CCC(CNC(=O)COCC1CCCC1)C(=O)N1CCCCCC1 C1(CCOC)(NC(c2ncc(C(F)F)s2)=O)CCN(C(c2sc(C)cc2C)=O)C1 C1(CNC(c2cc(CC3CC3)on2)=O)CC(O)CN1C(=O)CC(F)(F)F N1(C(c2cc(C)[nH]n2)=O)CC2CCN(C(=O)Cc3cc(Br)ccc3C)C(C2)C1 c1(C(N2C(C(C)NC(c3c(C)cccn3)=O)CCC2)=O)nc2c(s1)CN(C)CC2 C(=O)(C(C)C(C)(F)F)NCC(C)CN(C)C(c1cc(I)c[nH]1)=O C1(c2n(CCC)nnn2)(NCc2ncc(CCC(=O)O)[nH]2)CCCCC1CO c1(CC(=O)NC(C2CCN(C(=O)Cn3cc(C#N)cn3)CC2)C)ccc(O)nc1 c1(C(=O)OC)c(NC(=O)C(C)N(C)C)sc2c1CCC(C)(C)C2 C1(NC(CC2CC(OCC)C2)=O)CN(C(C2C=CCS2)=O)CC1SC CC(N=c1nc(Br)[nH]s1)C1CC2(CCCCC2)C1 C(=O)(C1=CCCC(C)(C)C1)N1CCCN1.c1(C(=O)OC)ncccc1Cl c1(C(N2CC(CN(C)C(C3CC4CC3C4)=O)OCC2)=O)cnc2[nH]cncc1-2 c1(C(N2CC(C(N(CC)CC)=O)OCC2)=O)cc(Cl)cn1C Cc1ccc(C=CC(=O)NCCCCC2(NC(c3ccccc3C)=O)CC2)o1 N1(C(CC(COC)C)=O)CCC(O)C(NC(C2CC(CF)C2)=O)C1 C1(OCCNC(C(CC)OC)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 N1(C(=O)OC(C)(C)C)CC(NC(c2cc[nH]c2C2CC2)=O)C(C2CC2)C1 N1(C(c2c(C)cn(C)n2)=O)CC2CCN(C(C3CNC(=O)CC3(C)C)=O)C2C1 C1(CNC(=O)Cc2ccco2)CN(C(c2cncc(-c3ccoc3)c2)=O)C2CC12 c1(NC(c2cccnc2S)=O)ccc2c(c1)CN(C(=O)CC1(O)CCOCC1)C2 N1(C(c2[nH]cnc2C)C(=O)NCCC)CCOC(c2ccc(Br)cc2)C1 C(C)(C(=O)N=c1ccn(CCO)[nH]1)N(C(CC1CC(OCC)C1)=O)C1CC1 N1(C(C(OC)OC)=O)CCOC(CCCC2CCCN2C(C2CCOC2)=O)C1 N1(C(c2c(C)cccn2)=O)CCC2C(CCN2C(c2[nH]nc3ncccc23)=O)C1 C1(CN=[N+]=[N-])CCN(C(C2(NC(C3CC(OCF)C3)=O)CCOC2)=O)C1 C(C)(C(C(=O)NC(c1nocc1C(=O)NC(CO)C1CC1)C)N(C)C)OC N1(C(CN(CC#C)C(c2ccc(OC)s2)=O)=O)CC2CC(C)C2C1 C12(CNC3CN(C(=O)Nc4ccoc4)C3)COCC(c3ccccc3)(C1)C2 C1(NC(C(C=CC)O)=O)CCC12CN(C(c1cnc(Cl)[nH]1)=O)C2 C1(C(=O)NCC2N(C(c3nc(C)nn3C)=O)CCOC2)CC2CC(O)CC(C1)C2 C1(NC(CC2(C)CC2(F)Cl)=O)CCCCN(C(C2(Cc3cccnc3)CC2)=O)C1 N1(C(c2ccc(CC)cc2OC)=O)CCN(C(=O)C(C)(O)C(C)(C)C)CCC1C Cc1ccc(N(C(=O)CC2C=CC(NC(C3(O)CCSCC3)=O)C2)CCO)cc1 c1(NC(CCC=CC)=O)ccc(NC(c2cc(Cl)cnc2O)=O)cc1C c1(C(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2O)ccc2cc(Cl)ccc2n1 c1(C(=O)NCC(CC=C)NC(C2(CO)CCCO2)=O)cc(S(C)(=O)=O)cs1 c1(CC(N2CC(NC(=O)C=CBr)(CO)C2)=O)ccc(Sc2cccc(Cl)c2)cc1 C(=O)(CC1=CCN(C)CC1)N1CC(C(C)C)N(C(c2cnn3c2CCC3)=O)CC1 C1(NC(=O)CC2CCC3CC23)CCN(c2nnco2)C12CCCC2 N1(C(C2C(OC(C)=O)C2)=O)CC2CC1CN2C(=O)C(C)=C(C)C CC1CCN(C(C2CC3CCC2O3)=O)C1CNC(c1cc(C(C)(C)C)ccn1)=O C(=O)(CCCC(=O)NCCCCNC(=O)C(c1c(C)noc1C)C)OC N1(C(C(CC)C)=O)CCCC2(CCN(S(=O)(=O)c3ccc(Br)cc3F)C2)C1 c1(C(N2C3C(NC(C4(COC)CC=CC4)=O)CC(C3)C2)=O)cc2n(c1)CCOC2 C12(CC)CC(C(=O)NCC3(C)CCN(C(=O)C4=CCSC4)C3)(CO1)C2 N1(C(C2CC3CC3C2)=O)CCC2(CCN(C(C3(C4(O)CCOCC4)CC3)=O)C2)C1 N1(C(CCCOC)=O)CCN(C(c2ccnnc2)=O)CC1C(C)(C)C c1(C(=O)NC2CCCC2NC(C2(F)CC3(CCC3)C2)=O)c(OC(F)F)cccc1Cl C1(C(=O)Nc2c(OCC=C)cccc2)CN(C(=O)CCSC)C2(CCCOC2)C1 Cc1cc(C(=O)NC2CC(CNC(c3cccc(OCC(F)F)c3)=O)C2)cn1C c1(C(=O)NC2C(C(=O)NCCCCC=C)C2)ccc2cccnc2c1 CC12CC(NC(=O)Cc3cncnc3)(C1)C1(CN(C(C3C=CCCC3)=O)C1)O2 S(=O)(=O)(c1ccc(C(=O)NC(=O)OC)c(Cl)c1)NCCC(C)NCC(F)F N1(C(C(n2ncc(C)c2)C)=O)CCC2CN(c3ccnc4ccnn34)CC12 c1(C(N(CCNC(C(C)n2ccnc2)=O)CCOCCO)=O)ccc(F)c(O)c1 Cc1cc(N)n2ncc(C(N3CC4(NC(C5CCCC5)=O)CCC3CC4)=O)c2n1 N1(C(C2C(C)=CCC=C2)=O)CC2(CCCC2NC(c2ccnnc2O)=O)C1 C1(C(N(C2COCC2(C)C)C)=O)CC(C)(C)CN1C(C1CC2CCC(C1)C2)=O C(CC(F)(F)F)(C(F)(F)F)NC(C(=O)N(c1cnc(N(C)C)s1)C)=O N#Cc1cnc2c(F)cc(Cl)cc2c1N1CCCC(C2CC2NC(=O)CSC)C1 N1(C(C(C)N(CC)CC)=O)CCC(C2CC2)(NC(c2cc(CC)n(C)n2)=O)C1 N1(C(CCc2onc(C)n2)=O)CC(CC(N2CCN(C(C)=O)CC2)=O)CC1(C)C C(=O)(CS(=O)(=O)c1ccccc1Cl)N1C(C)CCN(C(CSCC)=O)CC1 C1(OCC)CN(C)C(C)(C(=O)NC2COC2)C1.c12cccnc1NC2 Oc1c(CNc2cnc(-c3cnn(-c4ccccc4)n3)nc2)cccc1Cl C12(C(N3CC(OC)C(C(=O)NCCC4COCC4O)C3)=O)CCCC1OCC2 c1(NCCCCOC)cc(N2CCOC(c3ccccc3Cl)C2)nc(C)n1 C1(NC(C2CC(C(F)F)(OC)C2)=O)CCCCC1NC(c1cc(CF)nn1C)=O Cc1[nH]nc2ncc(N(C3CC4(CCNCC4)C3)CCS(=O)(=O)CCCCCl)cc12 CC1CCC(C(=O)NC2CCC2NC(c2ccc(CSCC(F)(F)F)o2)=O)O1 N1(C(CC(C)(C)n2cc(C(CN(CC)CC)C)nn2)=O)CCn2cc(C)nc2C1 c1(N(C(C23CC(NCc4cc(Br)cnc4F)(C2)C3)=O)CCO)cc(Cl)ccc1O N1(C(Cn2c(C)ncc2)=O)CC(NC(=O)CSc2ccccc2)C(F)(F)C1 n1(CC)nnc(C(=O)NCCN(C2CCCCC2)C(=O)CC2CCC(=O)N2)c1C N1(C(c2ncn(C)c2Cl)C(=O)Nc2c(C)c(Cl)ccc2)CCc2cccc(O)c21 Cc1nc(N2CCC(CC(=O)NC(C3(O)CCCCC3)C)C2)n(C)n1 Cc1nccc(N2CCC(OCCNC(=O)C(c3cccnc3)C)C2)n1 C1(NC(C(CC=CC)NC(C2CC23CCCC3)=O)=O)CN(C)C2(CCC2)C1 CC(Cn1cccn1)C(=O)NCCCC(=O)NCc1ccc(C(N)=O)o1 n1(CCNC(C2N(C(c3cncc(OC)n3)=O)CCC2)=O)ccc(O)nc1=O C#CC1(O)CC(C(N2CCC(C(C)NC(c3ccc(Cl)cn3)=O)C2)=O)C1 CCC(CC)C(C)C(=O)NCCC1CN(C(c2cc(C(F)F)[nH]n2)=O)CCCO1 C1(NC(C(CSC)NC(C=CCCCCC)=O)=O)CCc2n[nH]cc2C1 N1(C(C(CC=C)N(C)C)=O)CCC2CCN(C(c3ccoc3Cl)=O)CC2C1 C(COCCNC)NC(=O)NCCOCC1CC1.CC.COC c1(OC)ccc(O)cc1C(=O)N(CCCCN(C(=O)C(C)(C)SC)C)C Cc1cc(C(=O)NCCCCNC(c2ccsc2Br)=O)ncc1CO N1(C(C(CCC)NC(C)=O)=O)CC2CC1CN(C(c1c(CC)noc1C)=O)C2 N1(C(CCCC)=O)C(CC(=O)N(C(C)CC)C)C2CCCC12 C12(C(=O)NC3C(NC(C4CC(=O)NCC4)=O)CC3)CC(C1)S(=O)(=O)C2 C(c1ccc(F)c(F)c1)=C1CCC(NC(c2c(C)c(C(=O)O)ccc2)=O)CC1 N1(C(Cc2cn(C)nc2)=O)C2CCC1CN(C(C13CCCCC1C3Br)=O)C2 N1(C(c2cn(CC)nc2)=O)CCC2(NC(=O)C(=O)NNS(N)(=O)=O)CCCC12 c1(OCC)ncccc1Cc1ccc(C(N(C(CNC(=O)CC)C2CC2)C)=O)[nH]1 c1(OC)cnc(C(=O)NCC(F)CNC(=O)CS(N)(=O)=O)cn1 Cc1ccc(N)c(C(=O)NCC2CCC2NC(=O)C2=COCCO2)c1 C1(CC(=O)O)CC(O)C1(C)C.C(=O)(CCCc1ncco1)NC(C1CN(C)C1)C.C1CC1 c1(CSc2nccc(C(=O)NCC3(O)CCCC3)c2)ccc(-c2ccncc2)cc1 C1(CNC(C(COC)C)=O)CC2(CCC2)CN1C(C1CC2(CCC2=O)C1)=O N1(c2ccc(-c3ccc(C)o3)nn2)CC2(CN(C(c3ccc(F)cc3)=O)C2)C1 c1(C(=O)NC(C(C)C)CN2CCCCC2)ccc2c(c1)CN(C(=O)C(C)C)C2 C123CN(CC1CS(=O)(=O)C2)CC(=O)N3.n1(CC#C)cnc(Cl)c1SC(C)C C1(C(C)C)CN(C(=O)C2=NOC(C)C2)CCN1C(=O)Cc1cc(C(F)(F)F)n[nH]1 C(=O)(CCCn1cc(C2CC=CC2)nn1)NC1(C(C)C)CC1 Cn1cnc2ccc(C(N3CC(NC(=O)C4CC4)C(O)C3)=O)cc2c1=O c1(C(N2CC(NC(c3cscc3Cl)=O)C2)=O)ccc(N2CCOCC2)c([N+](=O)[O-])c1 CCCCC(CNC(=O)COC(C)CC)NC(c1csc(-c2cccs2)n1)=O CC1CCCC(CC(N2CCCC2Cn2cc(C3CCOCC3)nn2)=O)CC1 C1(C)(C(=O)NC(C2(O)CN(Cc3nnc(-c4ccco4)o3)C2)C)CC(C)(C)C1 Cc1cc(C(=O)Nc2cccc(C(F)(F)F)n2)c(C)n1Cc1ccncc1 c1(C(N2C(C(=O)NC(c3cnc[nH]3)C)CC3(CC3)C2)=O)n[nH]c2cccc(F)c12 c1(CN(CC(C)O)Cc2ccccc2)cccc2c1OCC(=O)N2 c1(N(C)C)ccc(C(=O)NC2(C)CN(C(c3[nH]ccc3C3CCC3)=O)C2)cc1 N1(C(c2ccc3sncc3c2)=O)CCCCC2(CCN(c3ncc(Br)cn3)C2)C1 C(C)(C)(C(=O)NC(C1CCCC1)CNC(C1CC1c1cn[nH]c1)=O)N(C)C Cc1c(C(=O)NC(C)(CNC(=O)C(C)CC(F)F)C2CCC2)cccc1F C1(CC)CN(C(=O)CC2CCC2)CCN1C(=O)CCSc1ccccc1Cl N1(C(c2c(C)scn2)=O)CCC(NC(C23COC(CF)(C2)C3)=O)C(F)C1 C(=O)(C(O)CC(N)=O)N1C(CCC(=O)NCCSC2(C)CCOCC2)CCC1 C12CCCN(CC1)C(=O)C2.c1(C(=O)NCc2c(CC)nco2)c(C)ccnc1C Cc1[nH]nc(CO)c1C(=O)NCC1C2CN(C(c3cnc(N(C)C)cn3)=O)CC12 c1(C(=O)Nc2scc(C(N(C)CC#N)=O)n2)cccc2c1oc1ccccc21 c1(C(=O)NCC2(NC(CS(=O)(=O)NC)=O)CCC2)nccn2nccc12 C(=O)(CC(F)(F)CS(C)(=O)=O)NC1CCCC(NC(CSC)=O)CC1 C#Cc1cccc(C(=O)NCCOC(C)(C)CNC(C2SCCC2C)=O)c1 C1(CNC(C=CC)=O)CN(C(c2ccnn2CC2CCC2)=O)CCC12CCOC2 N1(CCc2cn(CCC(=O)OCC)nn2)CCOC(C(=O)Nc2ccccc2)C1 c1(N(C)CCC2CC2)nc2cc[nH]c2c(=NC2CCC(=O)N(CCO)C2)[nH]1 c1(COC)ccccc1NC(C1(C(C)(C)C)CCOCC1)c1nnnn1CCF CC(CS(C)(=O)=O)C(=O)NCC1CC1NC(c1ccc([N+](=O)[O-])cc1)=O N1(C(=O)CN2CCCC2CC(=O)Nc2n(C)ncn2)CC2CC3CC2C1C3 O=C(CS(=O)(=O)CC(F)(F)F)NCCC1COCCN1C(=O)C(F)CC1CCCC1 N1(C(CCC(=O)N(C(C)C)C)=O)CCN(C(=O)C(CO)OC)CC1CC1CC1 c1(C(=O)Nc2cc(C)ns2)ccc2n[nH]cc2c1C.C12CN(CC1C)C2=O n1(CC)ncc2cc(C(=O)NCC3CC(CNC(C4(Cl)CC4)=O)CO3)cnc12 Cc1cc(O)ccc1CC(=O)NC1CC(N(C(=O)C(C)OCC2CC2)C)C1 C1(C)(CNCCNC2CCCCN(C(=O)OC(C)(C)C)C2)CCS(=O)(=O)CC1 C1(NC(CCCCC=CC)=O)CCN(C(=O)CCNc2ccccn2)CC1(C)C c1(C(=O)NCC(C)CNC(c2cc(O)nc(O)n2)=O)ccnc2ccncc12 c1(C(CN(C(C2CC(F)(CF)C2)=O)CC)O)cccc(C(F)(F)F)c1 C1(O)(C(=O)NC(C)Cc2nc[nH]n2)CCN(C(=O)CCNC(N)=O)CC1 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCCCC1CNC(=O)CC1CN(C)C1 Cc1cc(C(=O)NCC23CC(CO2)N(C(C2CC(O)C2)=O)C3)cnc1C(F)F c1(C(=O)NC2CCN(C(C3C(OC)C3)=O)C2)cc(O)nc(Br)c1 C1(CNC(C(C)OCC2CC2)=O)CC2(CO1)CN(C(C1(C)CS(=O)(=O)C1)=O)C2 Cc1scnc1NC(N1CC(CCNC(=O)CNC(=O)CC2CCCC2)C1)=O N1(C(=O)CSc2n[nH]c(O)n2)CCCCC1CNC(C1CC2CCC1C2)=O C12(CCNC(C(C)(C)SC)=O)CCC1CN(C(=O)C(C)(C)c1cc[nH]n1)C2 CN1CCOCC1C(=O)NCC1CCC(CNC(=O)CC2(C)CC(F)(F)C2)CC1 C1(CNC(C(C)OCC=C)=O)(CNC(=O)CC(C)F)CC1(F)F c1(C(C)C)ccc(O)c(C(N2CCC(C)(CCNC(c3cn(C)nn3)=O)C2)=O)c1 N1(C(C)C)CCOC(C(=O)NC2CC(N(C(=O)CCN3CCOC3=O)C)C2)C1 c1(C(C)N(C)CC2CC2C2CC2)ccc(N(C)C)nc1 c1(C(N2CCC(OC)(CNC(C3CCC34CCC4)=O)C2)=O)c(Cl)cncc1Cl N(C1c2ccccc2CC1NC(c1cc(=O)cc[nH]1)=O)C(C(CC)C(C)(F)F)=O N1(C(C(C)Sc2ccccn2)=O)CCC2(CCCC2NC(=O)CCC(C)=O)CC1 C1(NC(C2CC=C(C)CC2)=O)CC2CCC(C1)N2C(C1(C)CC(C(F)(F)F)C1)=O c1(C(C)(F)F)n[nH]cc1C(=O)NC1CC1NC(=O)Cc1csnn1 C1(F)(C(=O)NCC2(O)CN(C(c3c(C(C)C)ocn3)=O)C2)CCOCC1 Cc1c(C(N2CCCC(O)(CN(C)C(C3CCCO3)=O)C2)=O)[nH]c2ccccc12 Cc1ncc2ccc(C(=O)NCC(O)CNC(=O)CC(C)(O)C3CC3)cn12 N1(C(C2C(COC)CC2)=O)CCN(C(C2(NC(=O)N(C)C)CC2)=O)CC1 c1(CCCNC(N(CCOC)C)=O)cccc2ccn(C)c12.C12(C)CC1S2 C1(NC(C2(CCNC(C3NC(=O)OC3)=O)CCC2)=O)C2CCCOC12 C1(C(=O)NCC2CC(C(=O)NCC(C)OCCO)CO2)(CC)CC=CC1 N1(C(c2ccnc(C)n2)=O)CC(NC(=O)C(C)NC(=O)C2CC2)CC(O)C1 CC(C)C(F)(CNC(C1CCOC1(C)C)=O)C(=O)Nc1cccc(C(N)=O)c1F c1(OC)ccnc(C(=O)N(C(C)CNC(c2cnc(C(C)O)s2)=O)C)c1OC C(c1ccncn1)=CC(=O)NC1CC(CC(=O)NCC2(CO)CCOC2)C1 CC1Cc2cc(C(=O)NCC34CC3CN(C(c3cc(Cl)no3)=O)C4)ccc2O1 c1(CN2CC(CC(N3CC4C(C(=O)OC)C4C3)=O)C2)ccc(C)c(F)c1F C1(C2CCN(C(=O)C(CO)C(F)(F)F)CC2)(CNC(C2(C)CC2)=O)CCOCC1 Cc1cccc(C(=O)NC2COCC2NC(c2ccc(CO)o2)=O)n1 C(C)(C)(CCC(=O)N1CCCC(O)(CCNC(=O)C2=CCCC2)C1)OC N(C(=NCc1cn(C)cn1)N1CC=C(c2c(F)cccc2F)CC1)C(C=C)C c1(CC(=O)NC2CCCC(NC(c3nnn(C)n3)=O)C2)cc(Cl)ccc1Cl c1(CC)ncccc1C(=O)NC(C)CCC(=O)NCCNC(C)=O C(=O)(C1=CC2(CCOCC2)C1)N1CCN(C(CCc2cc(C)on2)=O)C(C)C1 c1(SC)ccc(CN(C(c2n[nH]c(C)n2)C(=O)NCCCF)C)cc1 c1(C(N(CC(=O)O)Cc2scc(C)n2)=O)cccc2cc(Cl)ccc12 N1(C(CC2CCC(=O)N2CCF)=O)CC2CCC(C1)N2Cc1cc(F)c(F)cc1Cl Cc1cc(F)ccc1C(=O)NC(C)CCCCNC(c1nc(O)nc(O)c1N)=O C1(C(=O)NC(Cn2ncc(C)c2)C(=O)O)(CN)CCCOC1 C1(C(NOCCN(C)C)=O)CCN(C(c2cc(Cl)cn2C)=O)C1C1CC1 N1(C(C23CC(C(C)(C)C)(C2)C3)=O)CCC(F)(CNC(=O)CC2CC=CCC2)C1 c1(N2CCC(CC)C2)nc(NCC2CCSC2)cc(C)n1 C(C(C(=O)NCC(C)(C)C1(O)CCC1)C(C)C)NC(C(=O)NC(C)C)=O CC1CCCC(C(N2CC(N(C)C(c3cnnn3C)=O)C2)=O)CC1 C1(CCC)CCCC1C(=O)N(CCC(=O)NCCc1ncc(C)o1)CC c1(CC(N2CC(C)C(NC(C3CCC(C(F)(F)F)C3)=O)C2)=O)ccc(O)c(F)c1 C(N=c1[nH]c2c(c(=NCc3cncc4c3CCC4)[nH]1)CCC2)c1nc(CC)oc1 Cc1cc(C)c(CC(=O)NC(C)C(C)NC(=O)CC2COCCOC2)c(C)c1 c1(C(=O)NC(CNC(C(C)n2ccnn2)=O)(C)C2CC2)cc2n(c1)CCCC2 c1(C(=O)NC2CCN(C(C3(C)CC=CCC3)=O)CC2F)ncc2n1CCCC2 C1(Br)(C(=O)NC2CC(NC(CC(C)n3cccn3)=O)C2)CC12CCC2 c1(NC(N)=O)ccc(C(=O)NCC2(NC(C34CSCC3C4)=O)CC2)cc1 C1(NC(CCNC(COC)=O)=O)CC(NC(=O)CN(C)C)C(O)C1 N1(c2cc3nc(n2)N3)CCC2(CCCN(C)C2)C1.C(O)(C(C)C)N(CCSC)C C1(CCNC(C2(COC)CC=CC2)=O)CN(C(C2C=CCCC2)=O)CCCO1 c1(NCC(CCOC)O)cnn(C2CC2)c1C.n1(CC=C)nnnc1C1(C)CO1 O(NC(=O)CS(C)(=O)=O)C(C(=O)Nc1n(CC)ccn1)C C1(F)(C(N)=O)CCCN(C(=O)Cc2cncnc2O)C1 C=CCCCCCCC(=O)N1CCC(CCNC(=O)C(C)(O)C2CCC2)C1 C(=O)(C(C)CC(=O)c1ccc(Cl)cc1)NCCC(C)NC(CCC)=O C#CC1(F)CCN(C(C2C3CCN(C(=O)CCCC(=O)N(C)C)CC23)=O)CC1 c1(C(=O)NC(CC)CN2CCCC2)conc1C(C)NC(=O)C=CCO N1(C(CN(C)CC)=O)CCCC(C)(C)C1CNC(=O)C(C)Cn1cccn1 C1(C(=O)NCCN(C(c2ccc(C(C)=O)[nH]2)=O)C)CCC2(CC1)CC2 C(=O)(C1=C(C)CCOC1)NCC(C1N(C(CC)=O)CCC1)(C)C CCC(C)C(CNC(=O)CCN(C(=O)Cc1cn(C)cn1)C1CC1)OC C1(C(N2C(CCNC(CS(=O)(=O)NCC)=O)CSCC2)=O)CCC(=O)N1C1CC1 N1(C(C(N)=O)=O)CCN(C(c2cccc(=O)o2)=O)CC1c1cccnc1 Cc1[nH]c(C)c(C(=O)NCC(C2CC2)NC(=O)CN2OC(C)(C)CC2=O)c1C c1(C(=O)Nc2cc(Cl)ncn2)cc2cc(-c3cccc4c3CCC4)cnc2[nH]1 c1(C(C(N)=O)NC(=O)CC2CN(C(=O)Cc3ccsc3)C2)cccnc1 C1(O)(CCNC(C=C(C)C)=O)CCN(C(=O)Cc2ccnc(Br)c2)C1 C1(C(=O)NCCOCC(N2CC3(CC3)CC2CO)=O)CC2CC1OC(=O)N2 c1(C(=O)NC2(CNC(C3C(OCC)C3)=O)CCCC2)cccn2nnnc12 CCCS(=O)(=O)CC(=O)N1CCC(C(C(C)C)NC(=O)CC=CC(C)(C)C)CC1 c1(CC(=O)NC(CN(C(c2cn(CC=C)nc2)=O)C)C)ccc2c(c1)CCCO2 C(=O)(CC(CC)CC)N1C(C)CCC1.c1(C(N(CCC)CC)=O)cccc(COC)n1 CC1OC2(C)CC1(C(N1CCC1CNC(=O)C(F)C1CCOC1)=O)C2 C1(CC(N2CC(=C(CNC(C(c3cnn(C)c3)C)=O)F)C2)=O)C2COCC12 N1(c2c(C#N)c(C)cc(C)n2)CCCC2(CCN(C(=O)C(F)(F)C(O)C(C)C)C2)C1 c1(OCCC(=O)OC(c2ccc(C)cn2)CN(C)C)cc(Cl)ccc1Cl CN1CCCC(C(N2CCN(C3CN(C(=O)CC4CCSC4)C3)CC2)=O)C1 C1(CC)C(C(=O)N(CCC(N)=O)CC)CCN1C(C1CCN(C)CC1)=O c1(C(=O)NCC2(O)CC(CNC(=O)Cn3ccnn3)C2)ccc(Cl)cc1 C(C(F)F)(C(C)(C)C)NC(CCN(C(c1n(C(C)C)ccn1)=O)C(C)C)=O C(C(C(=O)NCC(C)(C)C(F)F)C(C)(C)C)NC(COCC(=O)NC)=O C1(C(=O)NC2CCC2O)(CC)CN(C(c2c[nH]cc2CC)=O)C1 CCCC(C(=O)N1CCCCC(NC(=O)CCn2cc(Cl)cn2)CC1)C(C)C N1(C(c2cccc(OC)c2F)=O)CC2CCC(C1)N2Cc1cn(CC(C)C)nn1 c1(OC)nc(C(=O)NC(C)(C)CN(C)C(c2cn(C3COC3)nn2)=O)ncc1F c1(C(=O)NC2C(CNC(C(CSC)C)=O)C2)cc2occc2s1 C1(CNC(C(CC)OCC)=O)CCCCN(C(=O)C(F)(F)NC(=O)OC)CC1 C(=O)(C1=NNC(=O)CC1)NC(CCNC(c1cc(C)n(-c2ccccc2)n1)=O)C c1(C(N2C3C(NC(=O)Cc4cnccn4)CC(C3)C2)=O)cc2c(nn1)CCOC2 C(CC(=O)NC(C)(C)COCCCNC(=O)COCCNC(C)=O)SC C(CCCCCNC(=O)OCc1nnccc1CO)OCCC Cn1cc(S(N)(=O)=O)cc1C(N1CCC(NC(C2C3COCC23)=O)C(O)C1)=O c1(C(N(C(CNc2c(C(=O)OC)ccc(O)n2)C)C)=O)ccc(C)cc1[N+](=O)[O-] N1(C(C(CNC(C)=O)(C)C)=O)CC2(CCCN2C(c2ccc(C)nc2NC)=O)C1 N1(C(Cn2nc(C)oc2=O)=O)CCCC2(NC(c3ncncc3Cl)=O)CC2C1 Cc1nc(-c2nn[nH]n2)ccc1NC(C1CCCN(c2nccs2)C1)=O Cc1cncc(C(=O)NC2CCN(C(c3cc[nH]c3C3CC3)=O)C2C2CC2)c1C C1(CNC(C=CC(=O)OC)=O)C(C)CCCN1C(c1cc(OC)cnn1)=O N1(C(c2n(C)ccc2)=O)CC(NC(=O)CC(C)(C)C)CC12CCOCC2 c1(C(N2C(C(C)(C)O)CCC2)=O)ccc(F)nc1 c1(OCC(=O)NCC#CCNC(C2(C)C=CCC2)=O)ccc(F)cn1 c1(N(CC(=C)C)C)nc(=NCC23CCCCC2C3(F)F)[nH]c2c1CSC2 c1(C(=O)NCC2(C)CC(NC(c3ccoc3CC(N)=O)=O)C2)ccc(F)cc1F c1(C(=O)OCC2OC(C)=C(C(=O)OC)C2)nc2ccc(Cl)cc2n1C C1(C(=O)NC(C)CC(C)(C)C)(NC(CC=C)=O)CCCCC1 C1(C(=O)NC2CC(CCNC(C3(CO)CCCC3)=O)C2)CCc2nn[nH]c2C1 Cc1cc(C(=O)NCc2cnn(CC3CCC3)c2)n(CCO)n1 CCCC(C)(C)CC(=O)NC1CC(O)CN(C(C2(CCO)CC2)=O)C1 C(=O)(C(O)C(C)C)N(CCNC(C(C)OCCC=C)=O)C N1(C(C(CC)N2CCCC2=O)=O)CC(OC)CC1CNC(=O)CC(C)C1CC1 c1(C(=O)NCCNC(CCOc2ccc(OC)cc2)=O)ccc2[nH]c(=N)oc2c1 c1(N(C(CC)C#N)CCOC)ccccc1CNC(C1(CC)CCOCC1)=O C(c1ccc2[nH]ccc2c1)=CC(=O)NCC(C(C)(C)O)F C1(NC(c2ccnnc2O)=O)CN(C(c2ncccn2)=O)CC1F Cc1ccc(C(N2CCC(CCC(N3CCC(C4(C)N=N4)C3)=O)C2)=O)c(C)c1 C1(O)(CNC(=O)CC2COCCO2)CCCN(C(c2cc(Br)ccc2Br)=O)C1 CC(C)C#CC(=O)N(CCCn1cc(C2C3COCC23)nn1)C1CC1 C(=O)(C(C(=O)OC)OCOC)NCC.C(CC(=O)NCCOCCC1CC1)SCC#C c1(OC)ccc(OC)c(C(=O)NC2CC(NC(=O)C=CC3(C)COC3)C2)n1 N1(C(C=CC=CC)=O)CCC(O)(CNC(c2cn(C)nc2CC)=O)C1 n1(CC(=O)NCCN(C(=O)CCc2ccc(Cl)cc2Cl)C)cc(F)ccc1=O c1(C(N2CCC3(CC2)CC3(F)F)C(=O)NC(C)(C)C)cc2c(cc1Br)OCO2 C1(CC(N2CCCC(n3cc(C(CCC)=O)nn3)C2)=O)CCC2CC1C2(C)C N1(C(C(CCC#C)NC(C2CCC(C3CC3)C2)=O)=O)CC2(C)CCC2(C)C1 C=CC(C)C(C)C(=O)NCC1(F)CN(C(=O)C(C)(C)C2CCOCC2)C1 c1(-c2nc(CN(C=O)CCCC3CC3(Cl)Cl)on2)ccc(F)cc1 c1(N(C)C)nc2ccc(NC(N3CC(N(C)C)CC4(CC4)C3)=O)cc2s1 c1(C(=O)NC2(CC)CN(C(c3cnc(OC)c(C)c3)=O)C2)cc(C)c(C)nn1 Cn1cc(C#N)cc1C(N1CC(O)CC1CNC(c1ccc(C2CC2)cn1)=O)=O c1(NC(C(CC2CCCC2)NC(C(C(=O)OC)OC)=O)=O)cnc2ncnn2c1 c1(C(=O)NCC(C)(C)NC(=O)Cc2cccs2)ncc[nH]c1=O C(=O)(C(C)S(N)(=O)=O)N1CC(OCCC(=O)NC2(C(C)O)CC2)C1 Cc1cc(C(C)C(N2CCC(O)(CNC(=O)COC3(C)CCC3)C2)=O)cc(C)c1 c1(-n2cc(C(CC)(C)NC(=O)CNc3ccccc3)nn2)ccccc1CO O=C(CC1OCCc2ccsc21)NCC(O)CNC(c1c[nH]c2ccccc12)=O N1(C(C(C(C)O)N)=O)CC(C(=O)Nc2ccc(C(=O)N(C)C)cc2)CC12CCC2 c1(OC)nc(C(=O)NC(C2CCN(C(=O)C(C)S(N)(=O)=O)CC2)C)cc(O)n1 N1(C(c2cc(C(C)=O)cn2C)=O)CCC(F)C(NC(=O)CN2CCC(O)CC2)C1 c1(C(=O)NCC2(F)CCN(C(C3CCCOC3)=O)C2)cc(F)cc([N+](=O)[O-])c1 N1(C(CCS(C)(=O)=O)=O)CCC2(C1)CN(C(C1CCC(N=[N+]=[N-])C1)=O)C2 N1(C(C(C=C)CC)=O)CCC(C)(C)C(CNC(=O)CCSC(F)(F)F)C1 C(=O)(CC(CCC)NC(=O)C(=CC1CCCC1)C)NCCc1onc(CC)n1 C1(CNC(C2C(C)C2C)=O)CC2CCC(C1)N2C(c1ccc(Cl)c(N)c1)=O C1(NC(CCCc2[nH]c(=N)sc2)=O)CC2CC(NC(=O)CCSC(F)(F)F)C1C2 n1(C(C)CC(=O)NC2CN(C(C34CCC3C4)=O)C2)c(=O)oc2ccccc12 Cc1cnc(C(=O)NCC2(C)CCN(C(c3cscc3C3CC3)=O)C2)cc1C#N Cc1oc([N+](=O)[O-])cc1C(=O)NCC1CC(O)(CNC(C2C3CCCC23)=O)C1 c1(C(=O)NC2(C)CC(NC(Cc3c(C)nsc3)=O)C2)n[nH]c(C2CC2)c1C N1(C(CC2CC(=O)NC2)=O)CC(NC(C2CN(CC(F)(F)F)C2)=O)C2(CC2)C1 C(CCC(C(=O)NCCc1ccccc1)NC(c1c[nH]c(C)c1)=O)OC C1(C(N2CC(C(C(=O)NCCN(OC)C)OC)C2)=O)CCC(=O)NC1 CCC(C)CCCC(=O)NC1(CCC(=O)NCC(O)Cn2cccn2)CCC1 c1(-n2ncc(NC(C)=O)c2)c(Cl)cccc1Cl.C12CN(CC1N1CCCC1)C2=O c1(C(N2CC(O)(CN(C(C3CC(C)OC3)=O)C)C2)=O)cccc2c1CCS2(=O)=O Cc1onc(Br)c1C(=O)NC(C)CCN(C)C(c1ccccc1F)=O C1(CC#C)(C(=O)NC(CSC)CC)CCN(C(c2scnc2Cl)=O)C1 C1(NC(c2ccc(Cl)c(Cl)c2)C(=O)OC)CC2CNCC2(c2ccccc2)C1 C1(N(c2cncnc2)C)COC2(CCN(C(=O)C(Cl)Cl)CC2)C1 Cc1nc(C(N2CC(CNC(c3csc(CO)n3)=O)C(C)C2)=O)c2ccccn12 CCC(CC(C)CO)NC(=O)CCCCN(C(=O)CCC1(C)CC1)C Cc1ccc2c(c1)N(C(c1coc(CNC(=O)COCC3CCOC3)n1)=O)CC2 N1(C(c2ccc(CCCC)cc2)=O)CCCC2CN(C(=O)CCC(C)OC)CC12 C(C(CC(=O)NC(C)(CO)C(C)C)NC(=O)C=CCN1CCCC1)OC CS(=O)(=O)c1ccc(F)c(C(=O)OCc2cc3n(c2)CCC3)c1 c1(SC)cccc(C(N2CC3CC3(NC(C3CCCO3)=O)C2)=O)c1Cl N(C(=NCCCF)NC(c1ccoc1)C)CC(C1CC1)OCC c1(-c2c(C(N(CC(C)CNC(C3(C)C=CCC3)=O)C)=O)c[nH]n2)ccccc1Cl N1(C(c2c(C)n(C)cn2)=O)CCN(C(=O)CCCNS(C)(=O)=O)CC(O)C1 C(=O)(C(C)(C)C(=O)NCCNC(=O)CCSCc1ccccn1)OC C=CCC(C)(O)C(=O)NCC(CC(C)C)NC(=O)COc1cc(C)cc(C)c1 N1(C(Cn2ccc(C)cc2=O)=O)CCC2C(NC(c3ccc[nH]3)=O)C2CC1 S(=O)(=O)(c1cnc(NC(C2CC(C#N)C2)C)c(Cl)c1)Nc1cccc(C2CC2C2CC2)c1 C1(C(=O)NCC(CNC(C2CCS2(=O)=O)=O)O)SC2C=CC1CC2 Cn1cnnc1S(=O)(=O)NCCNC1CCCC(F)(F)C1 c1(C(=O)NC(C)C(C)(C)NC(=O)C(F)C2CCC2)cc(F)ncc1Br CCC(CC)C(=O)N1CCN(C2CCN(C(=O)CCC3CCCCO3)C2)CC1 C1(C(N)=O)CCC(NCC2CC3CCC2O3)CN1 N1(C(c2c(SC)ccs2)=O)CC(CNC(C2C3CC4C(C3)C24)=O)C(O)C1 N1(C(C23CCC(OC)C2C3)=O)CCC2(C1)CN(C(c1cc(F)ccc1Cl)=O)C2 c1(C(C(=O)NCCCF)N(C2CCCC2)CCc2scc(C)n2)cnccc1C C1(C(F)(F)F)(NC(C)=O)CCN(C(c2csc(I)c2)=O)CC1 C(=O)(CC(C)CC(C)C)NC(CC#C)CC(=O)NC(c1nc[nH]n1)C1CC1 C(=O)(C#CC1(C)COC1)N1CCN(C(CC2(C(=O)OC)CCSCC2)=O)CC1CF Cc1cc(O)ccc1C(=O)NCC1CCC1NC(=O)C(C)(C)C1CCCCO1 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCC(C)(NC(c2ccc(C)cc2)=O)C1 CC1(C)CC(CC(=O)NCCC2CC2)N(C(C2CC(=O)CCO2)=O)C1 c1(CCNC(COCCNC(=O)CCSC2CC2)=O)cccc(O)n1 C1(C(=O)NCCN(C(CC)C)C)(N(C2CC2)CC)CCc2cc(Br)ccc2C1 c1(CC)ncc(Cl)c(C(=O)NC(C)CCCNC(c2sc(=N)[nH]c2C)=O)n1 c1(OC)ccc(C(C(F)(F)F)NC(=O)CCSCCC(C)(C)C)cc1OC N1(C(CSC)=O)CC2CCOC2(CNC(c2n[nH]c3c2CCOC3)=O)C1 C(=O)(C=CS(C)=O)N(C1CCN(C(=O)CCc2cncc(O)c2)C1)C N1(C(c2n(CCC)ncc2)=O)CCC2(CCN(C(=O)C(C)NC(N)=O)C2)C1 C(=O)(CCCCCN(C)C)NC(C(C)(C)NC(c1cccc(CC=C)c1)=O)C C1(Nc2cccc(NC(C3OCCN(C(C)=O)C3)=O)c2)CCc2nc(C)[nH]c2C1 c1(CN(C(c2cn(CC#C)nc2)C(=O)NCC2CCC2)CC=C)ccccc1Cl C1(C(N(CCC(=O)NC(C2CCCCC2)C)C)=O)CCCSC1C c1(CC)ccnc(C(=O)NC2CCCC(CNC(=O)CCC3CCOC3)C2)c1 O=C(C#CC1CC1)NCc1c[nH]nc1C(=O)NC(c1cccs1)CO c1(CN2CCCS2(=O)=O)ccc(-c2nc(C(N3CC(CN)C3)=O)cs2)cc1F O=C1CN(C(CCC2CCCO2)C(=O)NCC2CCOC2)CCCN1 CC(C)CC(F)(F)C(=O)NCC1(C)CCCN1C(=O)CCN1CCOCC1=O c1(NC(C2CCN(C(=O)OC)C2)=O)ccc(NCCCc2ccsc2)nc1 c1(C(=O)NC(C)CCNC(=O)CSCc2ccncc2)[nH]cc2c1CCC2 C1(NC(CCCOC)C(=O)OC)CCCN1S(=O)(=O)N(C)C CC1=C(C(=O)NCCC(C(C)C)NC(=O)CC(c2c(C)noc2C)C)SCCO1 CC1Cc2ccccc2C1Nc1nccc(Br)c1C#N C1(C(N(C2CN(C(C(=Cc3cccs3)C)=O)C2)C)=O)CC(C)(C)OC1(C)C c1(C)nnc(N(C)CC)n1CCC1CCCCO1 c1(C(=O)NCCCNC(CC(C)C2CCCO2)=O)cc(Cl)c(F)cc1Cl c1(C(=O)NC2CCCN(C(COCCC(C)C)=O)C2)cc2occc2n1C c1(COCC)nc(N2CCCCC(CNCC3C(C)OC(C)C3C)C2)cc(C)n1 C=C(Cl)C(C)(C)C(=O)N1CCOC(CNC(=O)Cn2cc(C3CCOC3)cn2)C1 C1(NC(c2c(C)n(CC(F)(F)F)nc2)=O)CCS(=O)(=O)C(C)C1 C1(NC(C2C(C)(C)C(=O)NC2)=O)CC2(CCN(C(c3cc(C4CC4)no3)=O)C2)C1 N#CC12CC(C(=O)NCC3(NC(C4CC(F)(CO)C4)=O)CCOC3)(C1)C2 c1(CCC(=O)NC2C(NC(C(CN(C)C)O)=O)C2)ccc2ccccc2n1 C1(NC(CCc2scc(C)n2)=O)CCOCC1NC(c1cn(C)nn1)=O Cc1ccc(C(=O)NC2CC(C(N3CCCC3C)=O)C23CCC3)c(C)n1 c1(C(=O)NCC23CC(NC(C4CC(C)OC4)=O)(C2)C3)noc2c1COCC2 CC1C(NC(=O)C(C)(C)CN(C)C)CCN1C(=O)CC1CCC(=O)N1C CC(C)CC(C(=O)N(C)C)N(C(=O)CC1CCN(CC#N)C1)C Cc1ccc(C(=O)NC(CC2CC2)C(=O)NC2CC(CC(N)=O)C2)c(C)n1 N12CC(O)(C1)C(F)C(=O)NC1(CC1)C2=O.c1(C2C(CO)C2)cccnc1 c1(C(=O)NC(C(N2C(C)(CCC)CC2)=O)CO)ccncc1F C1(CC(=O)N(CCNC(c2ccc(CC)s2)=O)CC2CC2)CCCS1(=O)=O C(=O)(CC(C1CC1)NC(=O)CC1COCCO1)N(C1CCOC1=O)C N1(C(Cc2c(C)occ2)=O)CCC(O)(CN(C(=O)Cc2ccco2)C)CC1 CC1CC2CN(C(C34COCC(C3)C4)=O)CC2N1C(=O)Cn1cc(C#N)cn1 CC1(C)CC(NC(=O)CCC(=O)N2CCOCC2)CN1C(=O)C=C1CC1 C1(NC(=O)Cn2nccn2)CC2CC(C1)N(C(c1cc3cnccc3[nH]1)=O)C2 C=CCCC(F)(F)C(=O)N1CC(CNC(C2CCCCCC2)=O)C(F)(F)C1 N1(S(CCOC)(=O)=O)CCC12CCN(C(c1ccco1)=O)CC2 C1(NC(c2c(C)occ2)=O)CCC12CN(C(=O)CCS(C)=O)C2 CN=c1ccc(C(N2CC3(CC3)CC2CNC(=O)C=CC(C)(C)SC)=O)c[nH]1 c1(NC(C(C)NC(c2c(C)cn(C)c2)=O)C(C)C)nc2ccc(Br)cc2o1 C(=O)(C(C)(C)CO)NCCN(C(C)C)C(c1cnn(C(F)(F)F)c1)=O C1(C(=O)NC2CC(CO)C2)(NC(C(C)OCC2CC2)=O)CC(F)C1 C1(NC(c2c(C(C)NC(=O)CCCCNC(N)=O)noc2)=O)C(=O)NCCC1C CC1CN(C(c2cc(C(F)F)ccn2)=O)CC1CNC(c1c[nH]nc1Cl)=O C1(C(=O)NCCCN(C)C(c2cc(C(F)F)nn2C)=O)CCn2c(O)nnc2C1 c1(CNC(C(COC)O)=O)nc(N2CCC(C)(CO)C2)cc(NC)n1.C(C)(C)OC N12CC(CC1(C)C)CC2=O.c1(CC)ccc(OCC(=O)OC(C)(C)C)cc1 N1(C(CCNC(N)=O)=O)CC(NC(c2cc(Cl)cnn2)=O)CC12CCCC2 CCS(=O)(=O)CC(=O)NC(C1(C(=O)NCCn2cccn2)CC1)C C1(N(C(=O)CSCc2cccs2)C)CC2CC1N(C(=O)Cc1ccnn1C)C2 N1(C(CC2(C)CC2)=O)CCN(C(=O)COc2ccc(F)cc2)CC(O)C1 C1(C(N2CC3CC3C2)=O)Cc2nccnc2CN1C(C1CC1(F)F)=O Cc1cc(C(=O)NC2CCC(CCNC(C3(CCF)CC3)=O)C2)cc2nn[nH]c12 c1(C(=O)NCC2OCCN(C(Cc3cc(C)ncc3)=O)C2)cc(CO)ccc1C c1(C(N2CCCC(CCNC(C(CC)(C)F)=O)CC2)=O)c[nH]c2c(C)cccc12 CC1(CNc2ncc(F)cn2)CCCN(C(C2(C)CC2C(F)(F)F)=O)C1 C(CC(=O)NC(C1CCCCC1)CO)(C(F)F)NC(C1=C(C)CC1)=O C(C)(CC(=O)OC)(C(=O)OC)N1C(CCC)CSC1.N(C)(NC(=O)COC)C C1(C(N(C)Cc2c(C)cco2)=O)CCN(C(c2sccc2Cl)=O)C1C(C)C CCC1=NOC(C(=O)NCC(=C2COCC2(C)C)F)C1 c1(OCC)ccsc1C(=O)N(CC(CC)NC(c1cnc(O)o1)=O)CC C1(C(N2CCCN(C(CC3COCC(C)(C)O3)=O)CC2)=O)CCC2CCCCN12 C(C)(CCCC(=O)NC1CCCCC1C#N)NC(c1cnn(CC)c1C)=O n1(CC)cnc(C(=O)NC(C)C(C)NC(C2(c3cc[nH]n3)CC2)=O)c1 C(CCC(CCC)NC(=O)COc1ccc(Cl)cc1Br)NC(CCC=C)=O N1(C(C2CCN(OC)CC2)=O)CCCC2(CCCCC2NC(=O)C(C)N(C)C)C1 C1(O)(NC(C2C(C(C)NC(COCCOCC)=O)C2)=O)CCC1 N1(C2C3C(CCCC2)C(=O)CN(CC#C)C3=O)CC(O)CC1C(N)=O C(CC(CC)C(=O)N1CC(NC(=O)Cc2ccc(O)cc2)C(CC)C1)=CC N1(CC#C)CCN(C(=O)C=CCN(C)C(c2ncccc2O)=O)CC1=O CCCC(C(=O)N1CC(CNC(=O)C(c2ccccc2CC(N)=O)CC)C1)OC N1(CC(=O)NCCCN(C(=O)CC2CC(F)C2)C)CCCC1 C=C(Cl)CC(C(=O)N1CCC1(C)C(C)C)NC(=O)CC1C=CCC1 C1(O)(C(C)NC(C(C)SCC)=O)CCN(C(c2cc(CN(C)C)n(C)n2)=O)CC1 C1(C)(C(N2CC(C(C(=O)NCC(COC)C)O)C2)=O)CC(F)C1 c1(CC)ccc(C=CC(=O)OC(c2nc(COOC)c(C(F)(F)F)o2)C)cc1.FC.O CC(CC(=O)NC1CCCN(C(c2cn(C)cn2)=O)C1C)P(C)(C)=O C1(NC(c2cnc(C(F)(F)F)s2)=O)CN(C(=O)C=Cc2cn[nH]c2)CC2CC12 C1(n2cc(-c3c(C)nco3)nn2)CC2(C1)CC(O)C2.C12CCCC1(C)NC2=O C1(NC(COCC)=O)CC(F)(F)CC1NC(=O)C(C)(C)N(C)C c1(C(=O)NCCCN(C(Cc2ccc(C)cc2)=O)C)cnc(O)c2ncccc12 N1(C(CC(=O)NCC#C)=O)CC(=O)CC1C(=O)Nc1cnn(CCF)c1 Cn1nc(CNC(=O)CC2CC2CNC(=O)C(F)n2ccnc2)n(C)c1=O c1(C(=O)NC(CC)CNC(c2cncc(C)c2Cl)=O)ccc2c(c1)NC(=O)NC2 N1(C(CC(C)C(F)(F)F)=O)CCC2(CCN(C(=O)C(O)P(C)(C)=O)CC2)C1 Cc1ccc(C2(C(=O)NCC=CCNC(C3CC3c3cncn3C)=O)CC2)c(F)c1 c1(C(N(CC(O)CNC(=O)CCc2cccc(O)n2)C)=O)coc(S(C)(=O)=O)c1 C1(OC)COCCC1N1CCN(CC)CC1.C1(C=O)CCCN1CCC1CCCC1 C(=O)(C(F)C1=CCCCC1)NC1CCC(CNC(c2c(C)n(C)nc2)=O)C1 N1(C(CC2(C)CN(CC34CCCN3CCC4)C2)=O)CCc2ccc(F)cc2C1 C1(C)(C(=O)NCCCC(C)NC(c2ncnn2C2CC2)=O)CCC(F)(F)CC1 N1(C(COCC(=O)NCCOC(C)(C)C)=O)CCC(C2CCOC2)C1 c1(C(=O)NC(C(C)NC(CN(C(C)C)C)=O)C)cnc(N2CCCC2)nc1 C(CN=c1ccnc(CNC2OCCC2C)[nH]1)N(CCC)C(C)C C(C)(C)(CC(C)NC(C1(c2ccc(Cl)s2)CC1)=O)NC(C)=O c1(OC)cncc(C(=O)NCC(C)(C2CCC2)NC(c2cnnn2C)=O)n1 N1(C(C(CC(=C)C)C)=O)CCC(F)(F)C(CNC(c2ccsc2COC)=O)C1 c1(C(=O)NCC2C(NC(=O)Cn3ccccc3=O)COC2)ccc(Cl)c(Cl)c1O N1(C(C2C(C(C)C)N(C(=O)CSC(F)(F)F)CC2)=O)CC2CC(O)CC1C2 N1(C(CC2(C)OCCO2)=O)C(C(=O)NCCN2CCNC2=O)CCC1C1CC1 C(=O)(C1=NN(C)C(=O)CC1)NC(COC)C(=O)NC1(CCOCC(C)=O)CC1 C12(NC(C(C)c3cc[nH]n3)=O)CC(CNC(c3cnns3)=O)(C1)OC2C C1(NC(COCC(C)(C)C)=O)CCN(C(=O)CNC(=O)NC2CC2)C2CC12 C(CCC1CCC1)(C(=O)Nc1cncc(F)c1)NC(C(C)CO)=O O=S(=O)(c1ccc(NC2CCCCC2)c(F)c1)N1CC=CC(O)C1 C12(C(=O)NC3CCN(C(=O)Cc4ccno4)CC3CO)CCN(C1)S(=O)(=O)C2 Cc1nc(N2CCN(C34CC(C(=O)OC(C)(C)C)(C3)C4)CC2)ccc1[N+](=O)[O-] Cc1ccc(C(=O)NC(C(=O)NC2CCCCC2(C)C)C2CC2)cc1O C1(C(=O)NC(CCN(C(C(OC)OC)=O)C)C(C)C)CCC(C)(C)OC1 C1(CN(C)C(c2csc(CO)n2)=O)CCCCN1C(=O)Cc1nc(C2CC2)n[nH]1 c1(C(=O)NC2CC(NC(C(C)OC)=O)C2)nn(C)c(Cl)c1Br C1(NC(C(CC2CCC2)NC(c2c(CC)ncnc2)=O)=O)CCCCC12CC2 C1(C(=O)NC(C)CNC(C2Cc3cscc3C2)=O)CC2(CO1)CC(F)(F)C2 C#Cc1ccc(C(N2CC(OC)CC2CNC(c2nn(C)cc2C)=O)=O)cc1C C1(C(=O)NC(CNC(c2cccc(C(N)=O)c2)=O)C(C)(C)C)CCCCC1(F)F N1(C(C2(F)CCCN(C(c3ccc(CC)o3)=O)C2)=O)CCCC12CCOC2C N1(C(CCc2nc(C)sc2)=O)CCC(C)C(CNC(=O)C=CBr)C1 CN1CC(C)(C(=O)NC2CN(C(c3ncc(F)cc3F)=O)C(C)(C)C2)CCC1=O n1(CCC=C)c(N2CCC(c3cc(C)no3)C2)nnc1C(C)[N+](=O)[O-] Cc1[nH]nc2c(C(=O)NC3CCN(C(=O)Cc4cc[nH]n4)C3C)cccc12 c1(-n2cc(C(=O)NCCN(C(Cc3nnc(C)o3)=O)C)nn2)ccc(Br)cc1 N1(CC(=O)CCC(=O)NC2CN(C(C(C#N)=CC(C)C)=O)C2)CC2C=CC1C2 c1(NC(C2C3CN(C(COC(C)=O)=O)CC32)=O)ccc2nncn2c1 CC1C(NC(=O)Cn2nccn2)CCCN1c1ncc(I)cn1 c1(C(N(C)CC2CCC(NC(C(C)C3CC3)=O)CC2)=O)n[nH]c2ccc(Cl)cc12 CCCCCCCCCCC(=O)N1CCCC(C)(C)C1CNC(=O)CC(=O)OC N1(C(N2CCC(N3CCC(n4cnnc4)C3=O)CC2)=O)CCc2nnnn2CC1 C1(OC)CN(C(c2ccc(NC(C)=O)cc2)=O)CC1NC(=O)CC1C=CCCC1 Cc1nc(CCC(=O)NC2(C)CC(NC(C3CCCN3CC(C)C)=O)C2)cs1 N1(C(c2ccc(OC)c(F)c2)=O)CCCN(C(C2NC(=O)CC2C)=O)CCC1 CCC(CC)CCCC(=O)N1CCOCC1CC(=O)NC(Cc1cnc[nH]1)CO C1(NC(CN(CC)CC)=O)CC2CCC1N2C(=O)CNC(C)=O c1(NC(N(C)CCc2ccccc2F)=O)cc(F)c2cn[nH]c2c1 C(=O)(C(C)(O)C(F)(F)F)N1C(CC(=O)N(CC(CO)C2CC2)C)CC(O)C1 c1(NC(C2C(CNC(C(COC(C)C)(C)C)=O)OCC2)=O)ccc2occc2c1 N1(C(CSCCN(C)C)=O)CCN(C(=O)C=Cc2cnccn2)C(C(C)(C)C)C1 c1(O)ccc(F)cc1.C1CCCC1.C12CC1CNC(=O)CC1(CC1)C(=O)N2 C1(CC(=O)NCC(N)=O)CN(C(c2ccc(Br)cn2)=O)CCO1 CC1(O)CCCN(C(=O)CCC2CCN2C(C2C3CC4C(C3=O)C24)=O)CC1 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(NC(c2ccc(C)nn2)=O)CC1C CC1CN(C(C2(NC(=O)Cc3ccc(F)cc3)CC(CO)C2)=O)C(C)C1C C1(C(=O)NCC2CCC2CO)CC2CN(C(C34CCCN(CC3)C4)=O)CC2C1 C1(C(=O)NCC2(NC(C(CN(CC)CC)F)=O)CCOC2)CN(S(N)(=O)=O)C1 C1(C(=O)NCC(CC)CCO)CC12CCN(C(=O)CC1(C)CC1)CC2 N1(c2c(C(=O)O)cc(-c3cnoc3)cn2)CCCC2(CCNC2=O)C1 C1(CC(=O)NC(C(C)NC(C(C)NC(=O)OC)=O)CO)CCN(C(C)=O)CC1 C(=O)(C(C)(C)C1=CCSCC1)N(CC(C)NC(c1cnc(OC)nc1)=O)CC N1(C(C(CC=C)CC=C)=O)CC2(C1)CN(C(C1(C)C=CCC1)=O)CCO2 c1(C(=O)NC(C)CCNC(=O)C=Cc2cccs2)cc2cccnn2c1 C1(CCCC)CN(C(=O)C(C)n2ccnc2)CCN1C(c1cocn1)=O C(=O)(C1=CC2CCC(C1)C2)NC1C(NC(=O)C2=C(C(C)(C)C)CC2)CCC1 C12(NC(CCN(C)CC)=O)CCCC1N(C(c1occc1C1CC1)=O)CC2 C1(NC(CC(C=C)CC)=O)CCSC12CN(C(=O)C1=NNC(=O)CC1)C2 Cc1ccc(C(=O)NC(C)CCN(C)C(c2ccnn2C(C)(C)C)=O)nc1C C1(NC(c2c(C)con2)=O)CC(C)N(C(c2cccc(NC(C)(C)C)c2)=O)C1 C1(C(=O)NC(C(=O)NC)CC2CC2)CC(C)CN(C(c2ccc(O)nc2)=O)C1 CC1NC(=O)OC12CN(C(C1(CNC(C3CC3Cl)=O)CCCO1)=O)C2 c1(C(=O)NC2CC2CNC(=O)C(F)C2CCCC2)cccc2ccnn12 Cc1cn2cc(C(N3CC4(CCC4NC(c4cncc(F)c4)=O)C3)=O)ccc2n1 C1(CCN(C)C(c2ccc(F)s2)=O)CCCCN1C(=O)Cc1cn(C)nn1 Cc1nn(C)c2c(NCC34CCCN3CCC4)nc(N3CCC(C(N)=O)CC3)nc12 c1(C(N2CCCCC(NC(C3CC3C(F)F)=O)C2)=O)cc2ccccc2nc1O c1(NC(C2CCN(C(c3cc(Br)cc(Br)c3F)=O)CC2)=O)cc2nccn2cn1 N1(C(C(CSC)C)=O)CC(N(C(=O)C2=CCCCO2)C)C(C)(C)C1 N1(C(C(CC2CC2)OC)=O)CCC2CN(C(c3ncnc4c3CCC4)=O)C2C1 Cc1nc(CN2CCCC2c2ccccc2)sc1-c1cnoc1 Cc1coc(C(C)(C)C)c1C(N1CCCC(CNC(=O)Cc2n[nH]c(=N)s2)C1)=O Cc1cc(C(=O)NCCC2CCN(C(C3CCS(=O)(=O)N3)=O)C2)c(O)nn1 c1(C(CSC)(C)NCCCn2ccnn2)nnnn1CCC1(C)CC1 N1(C(c2ccc(NC)cc2Cl)=O)CC2COCCC2(NC(=O)CSC(F)F)C1 C(=O)(C(CCSC)NC(N)=O)NCC(C)(C1CC1)NC(CCC=C(C)C)=O C(CCCC(=O)NCC(C1CCN(C(=O)C=CS(C)=O)CC1)F)SC Cc1nccc(CCC(=O)NCC(C(C)C)NC(=O)Cc2c(C)n[nH]c2C)n1 Cc1cc(C(c2nnnn2C2(C)CC2)NCC2(CS(C)(=O)=O)COC2)cc(C)n1 N1(C(C2CCCC(C)(C)O2)=O)CC2(CCCC(CNC(c3ccon3)=O)O2)C1 c1(N2CCC(C)(NC(=O)C=Cc3ccc(Cl)s3)C2)ncnc2ccc(Cl)cc12 c1(CC(=O)NC(COCC)C)ccc(C(C)(C)C)cc1.C1(=O)C(=O)NCCN1 CCC(O)C(C)C(=O)N1CCN(C(=O)CCOC(C)C)C(CC(C)(C)C)C1 CC1CN2CCN1C(C(=O)NC1CCC(CCNC(=O)Cc3cnc[nH]3)C1)C2 N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CCC(NC(C2(CC3CC3)CC2)=O)C(F)C1 C12(NC(C3CN(C)C(=O)C3)=O)CCCC1N(c1ncnc(=N)[nH]1)CCC2 C#CCCCCCC(=O)N1CC2CCC1C(NC(c1cn(C)cn1)=O)C2 CCCCCCCCC(C)C(=O)N1CC2COCC(C1)N2C(C1CCCS1)=O C1(C(=O)NCC2CCN(C(c3c(C)n(C(C)C)nc3)=O)C2)Cc2ccccc2N1 C1(CCNC(C2CCCOCC2)=O)CCN(C(C2CSC2)=O)CC1 c1(C(=O)NC(CC=C)CNC(=O)CCNC(=O)CC)cc(F)cc(F)c1 c1(C(=O)NCC2CN(C(c3c(C)scc3)=O)CC2O)cccc2ncsc12 c1(CNC(C(CCC)N(C)C)=O)nnc2n1CC(C(F)(F)F)CC2 Cc1cc(C(=O)N(C(C)CNC(=O)CCCCCF)C)cc(C)c1 N1(C(c2cnc(OC)s2)=O)CC2CCCC2(NC(c2c(C)nn(C)c2F)=O)C1 C12(C(N3C4(CN(C(CNC(C(C)C)=O)=O)C4)CCC3)=O)CCC(C#N)(CC1)CC2 C(=O)(CC(O)C(C)(C)C)NCCCCCNC(CS(CC)=O)=O N1(C(CCCCCN(C(C(C(C)C)C(C)C)=O)C)=O)CCC2(COC(C)C2)C1 C1(CC(=O)NCC2CCCN(C(C3C=CC=CC=C3)=O)C2)COCCOC1 C1(CNC(C2CN(C)C(=O)N2)=O)C2CCC(C2)N1C(c1ccc(C(F)(F)F)s1)=O Cc1cccc(C(=O)NCC2CCC(C)CN2C(=O)CC23CCC(CC2)C3)c1O C(=O)(CC(C)(C)N(C)C(C1CC2(CC2)C1)=O)N1CCC(CC=C)C1 N1(C(C(C)SCCCC)=O)Cc2n[nH]cc2C1C(=O)N(c1cn(C)nn1)CC C1(CNC(c2c(NC)cccn2)=O)CN(C(=O)CCC2OCCO2)CC(C)(C)C1 C=CCC(C(=O)NC1(C(=O)NCC(O)CNC(N)=O)CCN(C)C1)NC(C)=O C(=O)(C(CCC(C)C)NC(=O)C(F)C(CC)CC)NCCCCCCC=C c1(CC(N2CCC(CNC(C3(SCC)CC3)=O)C2)=O)ccccc1S(C)=O c1(CC)cc(CNC(c2conc2C(C)NC(=O)CC2CCCN2C)=O)no1 Cc1cc(Cl)cc(C)c1C(=O)NCC1CCN1C(c1cnsn1)=O c1(N(C(CNC(C=Cc2cnc(C)nc2O)=O)C)C)nc2cccc(Br)c2o1 c1(NC(C(C)NC(=O)CC2CCOC2=O)=O)cnccc1CO C#CCCCC(C(=O)NC1COC(C)(C)OC1)N1CCCC1c1ccncn1 CS(C)(=O)=Nc1ccc(C(=O)NCC2CCCO2)s1 C1(NC(N2CCOCC2c2ncon2)=O)OCCOC1c1ccccc1 c1(NC2CC(CN(C)C)C2)ccc(S(=O)(=O)N2CCC3(C2)CC3(F)F)cc1Cl N1(C(CC2C(COC)C2)=O)CC(O)(C(C)NC(=O)CN2CC(C)(OC)C2)C1 C(CC1=CCN(C(C2CC2c2ccco2)=O)CC1)NC(c1c(C)ccnn1)=O Cc1cnc(C(=O)NC2CN(C(=O)Cc3cccc(F)c3)CC2F)cc1Br C(CCCC(c1nnnn1C)NCC1CC(OC(C)(C)C)C1(C)C)OCC c1(C(=O)NCC2(CNC(C3N(C(C)C)CCCC3)=O)CC2)snc2ccccc12 c1(C(F)F)ccc(-n2nc(C3CCCCC3)nc2C2CC23CCC3)cc1 c1(NC(C2CN(C(c3cccc(NS(C)(=O)=O)c3)=O)C2)=O)cc(Cl)c(F)cc1Cl CCC(CC(=O)NCCCCCN1CCN(C(=O)CC(C)(O)C2CC2)CC1)OC C1(C(N2C(CN(C(C(CC)OC)=O)C)COCC2)=O)CCC=CCCC1 C1(C(=O)NCc2ccc(SC)s2)CCCC(CN2CC3CC3C2)C1 c1(C(N2CC(C(N(CCC(C)C)C)=O)C(C)(C)C2)=O)cc2ccccc2o1 C(=O)(C(C(C)C)NC(=O)C(C)(C)C)N(CCCNC(C(C1CC1)OC)=O)C CCC(CC(=O)NC(CN(C)C)C(=O)N(C1CC2CCC1O2)C)C(F)F C12(NC(C(C)=C3CCC3)=O)CC3CCC(C1C2)N3C(c1cc(Cl)ccc1N)=O c1(CNC(C(N2C(=O)CCC2=O)CC)=O)cc2n(n1)CCN(C(=O)CCF)C2 C1(CNc2ccc(C=CC(=O)OC(CCCOC)C#N)cc2)Cc2nnc(C)n2C1 c1(C(=O)NCC2CC3(CN(C(c4[nH]c(=N)sc4)=O)C3)C2)cnc2c(c1)CCCO2 C1(C(=O)NC(c2nc[nH]n2)C2CC2)(CC)CCN(C(=O)C(C(C)C)n2cncn2)C1 C(N=C(NC1CCCC1)N1CCC(c2cccc(F)c2)C1)c1c(Cl)nsc1 C#Cc1ccc(OC)c(C(=O)NC2CN(C(=O)C(C)CF)CCC2C)c1 c1(C(=O)NCCC2(CNC(CCS(=O)(=O)NC)=O)CC2)nc(C)c(C)[nH]c1=O C(=O)(C(CCC(N)=O)NC(=O)OC(C)(C)C)Nn1ccc(C)cc1=O CCCC(O)(CNC1(C(=O)OC)CCNC1(C)C)C(F)(F)F C1(C(=O)NC2(COC)CCN(C(c3nc(O)c(C)s3)=O)C2)CCN2CCOCC12 c1(C(=O)NC(C2N(C(C(CC)O)=O)CCC2)(C)C)cccc(OC(F)F)c1 N1(C(C=C(C)C2CC2)=O)CCC2CCN(C(=O)CSCc3ccccc3Cl)CC12 C1(C(N(C2CCN(C(c3cnc(O)o3)=O)C2)CC)=O)CCCCC1(C)C c1(COC)ccc(C(=O)NC(CO)C(C)NC(=O)C(C)CC2CCCCC2)o1 Cc1cc(NC(CNC(c2cnoc2-c2ccco2)=O)C(C)(C)C)ncn1 O=C(CCCCCBr)NCC1CCCN(C(=O)CCCc2ccccc2Cl)CC1 c1(C(C)(C)C)nccc(=NC(=O)C2CCC(CNc3n[nH]cc3I)CC2)[nH]1 Cc1c(O)c(=O)ccn1CC(N1CCC(C)(NC(=O)Cn2cccc2)C1)=O c1(C(=O)NC(COCC)C(=O)NC(c2ccncn2)C)cccc(C)n1 C#Cc1ccc(C(=O)N(C2CCC(CNC(=O)C(C)CC(F)F)CC2)C)c(F)c1 C1(N(c2cccc(NC(=O)OC)c2)C(C2CCOC2C)=O)CCNCCC1C c1(C(N2CC3C(CNC(C4(CCCC)CC4)=O)C3C2)=O)cnc2occc2c1 C(CC(CC)C(=O)N1CCC(C(=O)NC2CCC=CCC2)(C(C)C)C1)=CC c1(OCC(=O)NC(CN(C(=O)C(F)C2CC2)C)(C)C)cc(Br)ccc1F C1(CC(=O)N(CC(CC)NC(C2CC2F)=O)CC)CCCN1C(C)=O.C(C)(C)(C)C(=O)O CC(O)CCCC(=O)N(C(C)CCNC(=O)C(C)(C)Cc1cnn[nH]1)C C(=O)(C1=C(C)N2CCN=C2S1)N(C1C(CC)CCCC1)C c1(C(c2n(CCCSC)nnn2)NCc2cnc(Cl)s2)cccc(C(F)F)c1 C=CCC(CC(C)C)C(=O)NCCOC1CN(C(=O)CCC(C)CN(C)C)C1 CC(C)CCC(=O)C(=O)N1CCN(C(c2ccc(CCO)cc2)=O)CC1C N1(C(C(C)(C)OCC)=O)CC2CC(NC(c3ccc(CC4CC4)s3)=O)C(C2)C1 c1(C(N2CC(CC=C)(NC(C3CC3F)=O)C2)=O)cnn(-c2ccc(O)nn2)c1N C1(C(N(CCC)CCC)=O)CC2(C1)CC(CO)C2.C1=CC(=O)N2CCC1CC2 C1(C(N(CCOC)CCNC(=O)CSCC(N)=O)=O)CCOCC1(C)C n1(CC)cc(CN(C(=O)C(C2CC2)N(C(=O)CC2CCC(C)C2)C)C)cn1 C1(CC)CN(C(=O)COCCCOC)CCN1C(c1cn(C(C)C)cc1C)=O c1(CN2CCCC(C(N3CC(C)C(O)CC3)=O)CC2)cc(F)c(Cl)c(Cl)c1 C(=O)(CCCCC#N)NC(CC)C(=O)NCc1cnn(C)c1O c1(CCC(N2CC(C)C(CNC(c3ccco3)=O)C2)=O)c(F)cccc1Cl N1(C(C=Cc2ccc(CC)o2)=O)CCC(C(F)(F)F)C(NC(=O)C(=O)NC2CC2)C1 C(C(CO)(CO)NC(C1CCC1c1nc(S)n[nH]1)=O)N(C)C(C1CCCC1O)=O CC1(C)CCN(CCNC(C2CC(Cc3cn(CCCC(=O)O)nn3)C2)=O)C1 c1(C(=O)NCC2CCN2C(C2CC3CC3C2)=O)cc2n(n1)CCO2 CCC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)C(CCSC)N(C)C)C1 C1(C(=O)NCCC(C)(C)NC(C(C)=C(C)C)=O)Cc2n[nH]cc2C(=O)N1 CC(O)CC(C)(C)CNC(=O)C(CCN(C)C)NC(c1ccc(O)c(F)c1)=O N1(C(CC(C(C)C)c2ccccc2)=O)CC2CCN(C(=O)C(C)(C)C)CC2C1 C1(C(=O)NC(CNC(c2cnc(CC)[nH]2)=O)(C)CO)CCC(=O)N(CC)C1 C1(NC(C(C)OC(C)(C)C)=O)CCCCC1CNC(=O)CSCc1ccccc1 CC1CCCCC1(CNC(C1CCCN1C=O)=O)NC(=O)CCn1ccnc1 Cc1cn2cc(C(=O)NC3CC(C)(NC(C4COCC(C)O4)=O)C3)nc2s1 CCCC(C)(O)C(=O)NC1CC(CC(N2CCC2CC)=O)C1 N12CCCC3(CCCCC3O1)CC(OC)=CC(C)=CC=CC2C(=O)NCC(F)F C(=O)(CCC(=O)c1cc(C)sc1C)NCC(CC=C)NC(c1cc(C2CC2)on1)=O C1(CNC(CC(=C=C)C)=O)CN(C(=O)C(CC2CCC2)OC)CC12CCOCC2 C=CC1COCCN1C(=O)NCc1oc(C)nc1C C1(C(=O)NCC2(F)CCN(C(=O)Cc3ccsn3)CC2)CC2C=CCC(C1)C2 c1(C(N2CCC(NC(CC)=O)C(CO)CC2)=O)ccc2c(c1)CCCS2(=O)=O CN1CCC(=CC(=O)N(C)CCNC(=O)Cc2cnc(C(C)(C)C)[nH]2)CC1 c1(C(N2CC(NC(=O)NC)C2)=O)coc(CNC(=O)CC2CCOC2C)n1 N1(C(c2cccc(C(=O)OC)n2)=O)CCc2ccc(-c3cnc(C)s3)cc2C1 c1(C(N2CC(CNC(c3c(C)ccs3)=O)C(O)C2)=O)cc(N)c(O)c(F)c1 N1(C(c2c(CC)con2)=O)CCC2(CO)CN(C(c3cnc(S)nc3)=O)CC2C1 N1(C(C2CC(C)(C(=O)OC)C2)=O)CCCC(O)(CNC(c2ccccn2)=O)C1 N1(C(c2c(C)csn2)=O)CC(CC(=O)NCc2cnc(O)c(F)c2)CC1(C)C C12(CNC(COCC(C)C)=O)CCCC1N(C(c1ccc(C#N)cn1)=O)CCC2 N1(C(c2c(C)scn2)C(=O)NCC(C)C)CCC2(CC1)COCC(=O)N2 Cc1ccc(O)c(C(=O)NC2(CNC(C34CCCC3C4)=O)CCOC2)n1 c1(NCCC2C(C)CCCN2C(=O)C2=CCCCO2)ncnc2cccnc12 C1(=CCNC(C2C(C)CCO2)=O)CCN(C(=O)C(F)(F)CO)CC1 N1(C(=O)NC(c2ccncc2C)CC)CCN(CC)c2c(F)cccc21 C1(C(=O)NCC2C(c3n(C)ncc3)C2)CC1C1CN(C(=O)CN2CC=CC2)C1 C12(CC(N3C(C)CC(NC(=O)C(F)=C4CCCC4)C3)=O)CCC(CC1)C2(C)C C1(C(=O)NC2CCC(NC(C3(CO)CCCCC3)=O)C2)CC12CCSCC2 C(=O)(C1=CNC2=NCCCN12)N1C(CCNC(C2CC(OC)C2)=O)CSCC1 C(=O)(C(O)CC(F)(F)F)N1CCC(N(CC#C)C(C2CC3(CC3)C2)=O)C1 C1(CNC(=O)CCCCO)CCN(C(C2CCCCC2O)=O)C12CC2 C1(CNC(C(C)Oc2cccc(Cl)c2)=O)CN(C(=O)CC(F)(F)F)CCCO1 C=C(C)C(C)(O)C(=O)NCC(C)(C(C)C)NC(c1cc2sccc2s1)=O Cc1nc2ccnn2c(C)c1C(=O)NCC(C1CC1)N(C(=O)CC1CCC1)C c1(C(=O)NCC2(F)CCC(NC(c3cc(C)n(C)n3)=O)C2)ncc(Cl)cc1Cl CN1N=C(CC(=O)NCc2ccc(CNc3ccnc4ncnn34)cc2)CC1=O N1(CC)CCC(C(=O)Nc2cnn(C)c2CS)CC1.C(C=O)=CCOCC.C1CO1 c1(OC)ccc(Cl)cc1C(=O)N(CC(O)CN(C)C(C1COCCOC1)=O)C C1(NC(CN(C)CCO)=O)CCC(CCNC(=O)CNS(=O)(=O)C2CC2)C1 C(=O)(C1=C2CCN=C2NC=C1)NCC1CC(NC(CN2CCC(=O)NC2=O)=O)C1 N1(C(CCSc2cccc(C)c2)=O)CCN(C(c2ccncn2)=O)CC1C1CC1 N1(C(CS(CC)(=O)=O)=O)CCCC2(C1)CN(C(c1csc(C(C)C)n1)=O)C2 C(=O)(C(F)CC(CC)CC)NCCC(C)(CC)NC(CC(CC=C)(C)C)=O Cc1nc(-c2cccc(F)c2)sc1C(=O)NCC(C)N(C)C(c1cnsn1)=O C(c1cc(C)no1)=CC(=O)NC(c1nc(CC(C)C)no1)C.C12(CC1)C(=O)NC2 C=CC1(C(=O)NC(CCC)C(=O)OC)CCN(C(C2CCOC2C(C)C)=O)C1 C1(C(N2CC(CC(=O)OC)(CC)C2)=O)CCC(C)N(C(c2cc[nH]c2OC)=O)C1 C1(NC(C(C2CC(NC(=O)CSC3CC3)C2)F)=O)CC12CCCC2 c1(CC)nn(C)c(CC)c1C(N1CCCC1CCNC(c1nc(=O)n(C)[nH]1)=O)=O c1(C(N(C)CC2(NC(c3cn(C)c(=O)cn3)=O)CC2)=O)ncc([N+](=O)[O-])n1C N12CCCN(CC1)CC2.O(N(CC1CCCCC1)C(=O)CC1CCCCCC1)CC c1(NCCNC(C)=O)cc(=NC2CCN(S(=O)(=O)C3CC3)CC2)[nH]cn1 c1cnc2c(=NCCC3CCCO3)[nH]c(NCCC3SCCS3)nc2c1 S(=O)(=O)(c1c[nH]c(=NC(CC)C2CC2)cc1C)N1CC(CC)S(=O)(=O)C(C)C1 N1(C(C2C(=C)C2)=O)CC2(CCC(NC(=O)CC3C=NN(C)C3=O)CC2)C1 C(C)(CCC(=O)N1CCN(C2CN(C(=O)CCCNC(N)=O)C2)CC1)OCC C(=O)(C(Cc1cccc(Cl)c1)=NO)NCC1CC(NC(C(CC)N(CC)CC)=O)C1 c1(CNC(C2(CNC(C(C)(C)c3cscc3Cl)=O)CC2)=O)cc(S(N)(=O)=O)c[nH]1 N1(c2cc(NC(c3nccc4n[nH]cc34)=O)ncn2)CCC2(CCCC2)C1 c1(C(=O)NCC(CC=C)NC(=O)C(O)C(F)(F)F)ccc2c[nH]nc2n1 C(=O)(CS(=O)(=O)CC)NC(C(=O)NCC(CCCC)O)Cn1cccn1 N1(C(C(C(C)O)C)=O)CCCC(C)(C)C1CNC(C1CC=CCO1)=O C1(CNC(C2CCCC3CC23)=O)COCCN(C(=O)Cc2ccc(F)cc2Cl)C1 c1(C(=O)NC2CN(C(c3nc(C)[nH]n3)=O)CC2C)cccc2c1C(=O)NC2=O c1(C(=O)NCC2(COC)CN(C(=O)C(C)(C)N(C)C)C2)cccc2c1ccn2C N1(CC(C)NC(C2(F)CCOC2)=O)CCN(C(=O)Cc2cnn(C)c2C(F)F)CC1 c1(N(C)C)ccc(C(=O)NCC2CC(F)CN2C(=O)CCCc2cccs2)cc1 N1(C(C(CNC=O)SC)=O)CCCC(NC(=O)COC2CCOC2)C1 CC1(C)CCC(C(=O)NCC2(F)CCOCC2)CN1C(C12CCN(CC1)C2)=O c1(C(=O)NCC(C)N(C)Cc2cc(C)on2)cccc2ncnn12 CC1CN(C(c2ccc(CF)cc2)=O)CCC1C(=O)NC(CO)CC(F)(F)F Cc1ccc(C)c(C(=O)NCCc2n[nH]c(=N)o2)c1O C1(C(=O)NCC(COC)(F)F)(CF)CCN(C(c2ccccc2CC#N)=O)C1 C(CC(C)C(=O)NC1CC(CNC(=O)CCc2c(Br)cnn2C)C1)=CC N1(C(C2CC(CC)(CC)C2)=O)CCCC(N(C)C(C2(C)CCCC2)=O)CC1 C(=O)(C1=CC2C=CC(C1)C2)NC1C(CNC(c2c(Cl)ccc(OC)n2)=O)CC1 c1(CNC(C2(CCCC)CCC2)=O)nc(C(=O)NC(C)CCCO)cs1 Cn1c(C(=O)NCC2(CCNC(C3CC(C4CC4)C3)=O)CC2)cc2ccccc12 CN1CC2CN(C(C3CCCCC3NC(C34C=CC(CC3)C4)=O)=O)CC2(C)C1 C(C(C(=O)N1CCC(F)(CO)CC1)C(C)(C)C)NC(C(n1ncc(C)c1)C)=O Cc1cc(C(=O)NC(C)CCCNC(=O)Cc2cnccc2Cl)n(C2CC2)n1 C1(N(C(CC)=O)C)CC2CC1N(C(=O)CC1OCCO1)C2.c12cccc(c1)CO2 C1(C)(COC)CCN(C(C2(CNC(c3cncc(C)n3)=O)CCCO2)=O)C1 c1(C(N2CCC3(CN(C(C(C=C)O)=O)C3)C2)=O)c(C)nn2cccnc12 CCC(CNC(c1ccccc1C(F)F)c1nnnn1C1(C)CC1)CCCO C12(C(=O)NC(c3ccccc3)C)CCC(CN(C(c3csc(C#N)c3)=O)C1)C2 c1(C(N2C(C3CCN(C(CCC(=C)C)=O)C3)CCC2)=O)ccc2c(c1C)CCC2 c1(OC)cccc(CN2CC3C(C2)N3C(n2ccc(CO)n2)=O)c1C c1(CC)ccc(C(=O)NC23COC(CNC(C4CCOCC4)=O)(C2)C3)cc1Cl C1(C(=O)NC(COC)CO)CCC(NC2CN(C(c3cc(C)n(C)c3)=O)C2)CC1 C(CN=c1cc(C)nc(Cc2cccc(C)n2)[nH]1)N(C(C1CCCSC1)=O)CC n1(CCCOC)cc(NCc2sncc2Br)cn1 C1(NC(c2c(CC(C)C)onc2)=O)CCN(C(c2nnsc2C)=O)C(C)C1 C1(OC)CN(C(=O)C(F)Cl)CC1NC(c1[nH]c(O)nc1C)=O C12(NC(c3c(CC)ccc(C)c3)=O)CCCC1CN(C(=O)C=CSC)C2 C1(CNC(c2cn(-c3cc(F)ccc3F)nn2)C)CC2(CO1)CC(C(=O)O)(CO)C2 N1(C(CC2C(C)C(=O)CC2)=O)CCC(NC(=O)CC2CC3CC3C2)C1(C)C C1(C(N2C(C(C)NC(C3CC(=C)CN3)=O)CCC2)=O)CCS(=O)(=O)C1 c1(OC)cccc(-c2nc(CC3CCSCC3)n(C(C3CCC3)C)n2)n1 N1(CCN(C(CC)=O)CC)CCN(CCc2cccc(OC)c2)CC1 c1(OC)nc(C)ncc1C(=O)NC1CCCCN(C(C2COC(=O)N2)=O)C1 CCCCC(CCCC)CC(CC)NC1CCCN(C(=O)OC(C)(C)C)C1 CCS(=O)CC(=O)N1CCCCC1CNC(=O)Cc1coc(C)n1 C=CCCCCCCC(=O)NC1C=CC(CNC(C2(O)CCCC(C)(C)C2)=O)C1 C(=O)(C(C)(C)C1=CCN(C(c2cccnn2)=O)C1)NCCCCCC(C)(C)C C(CN=C(NCC(=O)OC(C)=O)NCCF)C1(NC(CCNS(CC)(=O)=O)=O)CC1 C1(NC(c2c(NC(C)=O)cccn2)=O)CN(C(c2n[nH]c(C)c2O)=O)CCC1C C=CC(C)(O)CC(=O)N1CCC(CC)CC1.C1(=O)C(C)NC(=O)N1 Cn1ncc2c(N3CCC(C4CC4)C3CNC(C3CCCCS3)=O)ncnc12 C1(CNC(C(C)OCCOC)=O)CC2(CC(NC(c3csc(S)n3)=O)C2)C1 CC(C)(C(=O)N1CCCC(C(=O)NCCCc2ccccc2)C1)C(F)(F)F C(CCN(C(=O)CCCN(C)C(C)C)C)(C(C)C)NC(c1nc(COC)oc1)=O c1(C(=O)NC2CCCC(CNC(C(C)SCC)=O)C2)ccc(C)nc1O c1(CNC(c2n(C)nc(C3CC3)c2)=O)ccc2sc(C(=O)O)cc2c1 c1(C(N2CCCC(NC(C(C)(C)c3cccnc3)=O)C2)=O)cc(Cl)c(F)cc1N N1(C(CC(COC)COC)=O)C(C)CC2CN(C(c3cc(N)cc(F)c3)=O)CC12 C(=O)(CC1=NNC(=O)C1)NCC(C(C)(C)C)NC(c1cnc2n1CCS2)=O C1(CNC(c2cnc3n2CCC3)=O)CN(C(=O)C(F)CC2CCC2)C2(CCC2)C1 CCC(CC)(CCNC(=O)CCCCc1cnn[nH]1)NC(=O)C1=C(Cl)CC1 c1(OCC)cc(CN2CCC(C)(NC(=O)C(C)c3cccs3)C2)ccc1OC Cc1ccoc1C(=O)NC(CC1CC1)C(=O)NCC(O)Cn1cccn1 C(=O)(C(C)(C)C(=O)OCC)NCc1c(C(=O)NC(CC=C)CC)n[nH]c1 CC1CN(C(=O)C(C)(C)F)CC(C)CN1C(=O)CC1CCCN(C)C1 C(=O)(C1CCCc2nncn21)NCC1(CNC(c2ccc(C#C)cn2)=O)CCC1 C1(C(N(CC(=O)Nc2ccc(O)cc2F)CC)=O)Cc2ccccc2C1 c1(C(=O)NC2(CNC(c3c(NC)scn3)=O)CC2)c(Cl)c([N+](=O)[O-])nn1C N1(CC(=O)NC)C(=O)NC2(CCc3ccccc3C2)C1=O.c12cccc(c1CN)O2 C1(CCCNC(C(CN(C)C)O)=O)CN(C(=O)CC2CCC2)CCO1 C(C)(C(C(=O)NCC1CCOC1)NC(=O)CC1CCOCC1)OC N1(C(C)C)CC2C(C(N3CCC3C(=O)NC3CCC(c4nc[nH]n4)O3)=O)C2C1 Cc1cn2cc(C(=O)NC(C)C(C)NC(=O)CCc3nccs3)cc(C)c2n1 c1(C(=O)NCCN(C(C2(COCC)CC2)=O)C)cccn(C2CCC2)c1=O.C1(C)CC1 CC(C(=O)N(CC(C)(C)NC(c1cnc(C2CC2)nc1O)=O)C)C(F)(F)C(F)F CN(C)NC(=O)CCC(=O)N1CC(CNC(C2(O)CC(C)(C)C2)=O)N2CCC1C2 c1(C(N(CC(N2CC(OC)C(F)C2)=O)CC(C)C)=O)cc(C#N)n(C)n1 CC1(NC(=O)CC2OCCC2C(F)(F)F)CCN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1 c1(OC(C)C)cc(NCC2CCN2C(=O)CC(C)(C2CCC2)C2CCC2)ncn1 C1(C(=O)NCCCCCNC(C2ON=C(CC)C2)=O)Oc2ccccc2C1C Cc1cccc2cc(C(=O)NC3(C)CN(C(=O)CC4COCCO4)C3)cnc12 CC(F)(F)C(F)C(=O)N1CC=CC1(C)C(=O)NOCC1CCC1 c1(C(N2CCCCC(CNC(c3cc(F)n[nH]3)=O)C2)=O)ccc2cnccc2c1 c1(-c2cn(C(C)CNC(=O)C(C)C(=O)OC)nn2)ccc(C#N)cc1S(C)(=O)=O C1(NC(COC)=O)CN(C(=O)C=CC2CCCCC2)CC12CC2 Cc1ccc(CCC(=O)NC2CC(NC(=O)C(Cl)=CCl)C2)c(Br)c1 c1(NC(C2N(Cc3c(C)scn3)CCC2)=O)cccc(F)c1C c1(C(=O)NC2(CN(C(C(C)(c3ccccc3)OC)=O)C)CC2)ccccc1C C1(C(=O)NCC(CC=C)NC(c2cnnn2C)=O)CCN(S(N)(=O)=O)CC1 C(=O)(C#CC(C)(C)C)N1C(NC(=O)NCc2ccc(N(CC)CC)cc2)CCC1 c1(CCC(=O)N(C)CC2(NC(c3ccc(C)cn3)=O)CC2)ccc(F)cc1Cl C=CCCN=C(NCCC(C=CC(F)(F)F)OC)NC(C)CCF C(N=c1[nH]c(Cl)ncc1C(N)=O)C1N(C(CC(=C)C)=O)CCCC1C c1(CC)ccc(C(N2CC(NC(c3ccc(C#N)[nH]3)=O)CCC2C)=O)c(C)n1 C(=O)(C(=O)N=S(C)(C)=O)NC1C(NC(C2(C)CN(C)C(=O)C2)=O)CCCC1 N1(C(C2CN(C(=O)Cc3cscn3)CC2C2CC2)=O)CCc2c(O)noc2C1 N1(C(Cc2ccc(C)nc2)=O)CCCC2(NC(=O)C(F)C3CCC3)CC2C1 c1(C(=O)NC2C(C(=O)NCCCSC)CCC2)cccnc1O C1(C2CCCN(C(=O)C(C)(C)n3cnc(C)c3)C2)(NC(C2(CC)CCC2)=O)CC1 N1(C(c2c(CC)nc[nH]2)=O)CC2CCC1CN2C(C1CC1C(C)(C)C)=O CC(C)(CC1CC1)C(=O)NCC(C)(C1CCC1)NC(=O)CCN1C(=O)CCC1=O N1(C(=O)Cc2cnns2)CCCC2(C1)CN(C(C1CC=CC1)=O)CCO2 N#Cc1cc(N(C2CS(=O)(=O)C2)CCc2ccc(F)cc2F)nc(C2CC2)n1 c1(CC(=O)NCCCCC(C)NC(C2(C)CC2)=O)cc(Br)ccc1F N1(C(C2C(CCC)C2)=O)CCC(NC(C2(F)CCCC2)=O)C12CC2 c1(CC(=O)NCC2C(NC(CC=C(C)C)=O)CCC2)cnc2ncccn12 C(C(C)C)(C(O)C(=O)N1CC(CNC(=O)C(C)OC(C)=O)C2(CC2)C1)OC C(N=c1[nH]c(C)cc(=NCC(C)(C)OC(C)C)[nH]1)C1(CC)CC(C)(C)C1 N1(C(C2(CC)CNC(=O)C2)=O)CCC(C(=O)NC2CCOCC2C)CC1(C)C c1(CNC(C=C(C)C(C)C)=O)ccc(C(=O)N(C)CC2CCCO2)cc1 C1(CNCC)CCCN(C)C1=O.C(CC1CCC1)(C(=O)C(C(C1CCC(=O)N1)C)=O)N N1(C(C(=O)NC(CC)C)CC2CCO2)CCCC(c2ccnn2C)C1 C1(C(n2cc(-c3cn[nH]c3)nn2)C)CCCC=C1Br N1(C(CCCC2C(C)C2)=O)CCC2(CC2C2C3CCN(C(C4CCC4)=O)CC32)C1 N1(C(C2CCS2(=O)=O)=O)CC=C(CCNC(C23CC4CC2C3C4)=O)CC1 c1(C(N2CCCN(C(=O)OC)C(C)C2)=O)cc(OC)cc([N+](=O)[O-])c1 CC(C)(C)C(CC(=O)NC1CN(C(=O)CCP(C)(C)=O)CC1(C)C)C(F)F C#CCC(C)(CC)C(=O)N1CC(NC(c2ncc(Br)cc2F)=O)C(O)C1 C1(NC(C2C(C(C)C)C2)=O)CC2CCC(C1)N2C(=O)Cc1cnns1 N1(C(C(C2CC(F)(F)C2)OC)=O)CCSCC1CCNC(C1CCC=CCC1)=O N1(C(C2C(CC(C)C)C2)=O)CCN(C(c2cccc(O)n2)=O)C(C2CC2)C1 O=C(CC(=O)N)NC.c1(NC(C2CC2N2CC(C(N(C3CC3)C)=O)C2)=O)ccccc1 c1(CCNC(C(C=C)(C)C)c2nnnn2C)cc(OC)c(OC)cc1F c1(CNC(C2CC(OCCn3cc(CN(C)C)nn3)C2)=O)ncsc1S(N)(=O)=O c1(OC)cccc(CNc2csc(C3CCCO3)n2)c1Br C#CC1(C(=O)NCc2ccnn2C)CCN(C(=O)C(C)OC)C1 C1(C)(C(=O)OC)CCC1(C)C(=O)NCC(C)(C)CN(C(=O)C(F)C1CC1)C C(C(C)(C)CC(F)F)NC(C1CCC(C)N1C(c1cc([N+](=O)[O-])n[nH]1)=O)=O N1(C(CN(C(COC)=O)C)=O)CCCC(C(C)NC(=O)Cn2cc(CO)nn2)C1 Cc1nncc(C(N2CC(C3(NC(C4CCN4S(C)(=O)=O)=O)CC3)C2)=O)c1C c1(C(=O)NCC2CCN(C(=O)C=Cc3ncco3)C2)cc2c(cn1)OCCC2 Cn1cc2c(C(=O)NCC3CCCN(C(c4cc[nH]c(=N)c4)=O)C3)cccc2n1 c1(C(N2CCC(F)(CNC(C(C)SC)=O)CC2)=O)cc(=O)n2nccc2[nH]1 c1(C(N2CC(CNC(CCC#C)=O)C(C)C2)=O)c(Br)nc2n1CCOC2 c1(C(N(C2CCC(NC(CCSCCCC)=O)C2)C)=O)cc(F)cc2c1CCC2 C1(CNC(Cc2c(C)con2)=O)CC2CCC1N(C(=O)CC1CCC(C)CO1)C2 N1(C(c2nccc(OC)c2)=O)CCCC(O)(CNC(C2CC(C(C)C)=NO2)=O)C1 Cc1ccn(CCC(=O)NC2CC(C(C)NC(=O)CCCn3cccn3)C2)n1 c1(C(=O)NCCOCCNC(=O)C#CC2CC2)ncc(F)cc1F C1(C(N(C)C)=O)COC(C(F)(F)F)CN1C(=O)OC(C)(C)C.OCC N1(C(C(CCOC)NC(c2c[nH]nc2C)=O)=O)CC2(CCC1CO)CC2 CCCC(C(=O)NCC(C)(CO)NC(c1nn(CC)cc1Cl)=O)C(C)C c1(CC(C(=O)NC2CCN(C(C3C(C=C)C3)=O)CC2)C)ccc(F)c(F)c1 c1(C(=O)NC(C)CNC(C2(Cl)CC23CCC3)=O)ccc(P(C)(C)=O)cc1 N1(C(Cc2c(C)nsc2)=O)CCCC(C)(NC(C2CC=CCO2)=O)C1 C(=O)(C(CO)NC(=O)CC1CCC1)NCC1(OC(C)=O)CC1 C1(C(N(CCCCC#C)C)=O)CN(Cc2ccccc2Cl)CC1O c1(C(N2CC(C)(NC(C(C)NC(C)=O)=O)C2)=O)ccc(Cl)nn1 c1(C(=O)NCC2CC(NC(C3(C)CCNC3=O)=O)C2)cccc2cc(O)ccc12 C1(C(=O)NC2CC(NC(c3cc(F)cs3)=O)C2)CCc2ccnn2C1 C(CCCCC(=O)N(CC(C)(C)CNC(c1ccccc1N(C)C)=O)C)SC C1(CC)CC(O)CN1C(C1C=CCN(C(c2ncncc2N)=O)C1)=O C1(C(N(C(CC)CC)CC)=O)(NC(=O)CCN(C)CCO)CC(F)C1 C(=O)(C1=CCCCO1)N1C(C)(C(=O)NCCC2CCC(C)(C)O2)CCC1 C1(C(=O)NC2C(OC)CN(C(=O)CC3(C)CC3)C2)(OC)CCCCCCC1 c1(NC(C)(C)CCCF)ccc(S(=O)(=O)N2CCOC(c3ccco3)C2)cc1Cl c1(CCNC(c2n(CCCSC)nnn2)CC2CCC(C)(C)O2)ccccc1O Cc1c(C(=O)NCCC2C(C)CCCN2C(=O)CCC(C)C)cccc1F C1(COC)CCCCC1C(=O)NCc1csc(CNC(=O)C=CBr)n1 c1(OCC=C)ccccc1C(=O)NCCCCC(C)NC(=O)Cc1nc[nH]n1 n1(CC)nc(C(=O)NCC2COCCN(C(C3CCCO3)=O)C2)c2c1CCOC2 C1(C(N2C(CNC(c3csc(O)n3)=O)CCC(C)C2)=O)Cc2ccccc2N1 C1(Nc2c(CC(=O)N(C)Cc3ccc(OC)cc3)cccc2)CC2CCCC2C1 CC1CCN(C(c2cc(Cl)n[nH]2)=O)C1CNC(c1cnsc1)=O C(=O)(CCN=c1[nH]ccs1)NC(C1CCN(C(c2ccc(Cl)s2)=O)CC1)C CC(C)C(CCN(C(=O)C(C)NC(=O)Cn1cnnn1)C)NC(=O)C(C)(Cl)Cl c1(C(=O)NCC2=CCN(C(C(n3ncc(C)c3)C)=O)CC2)cnc2sc(C)cn12 c1(C(C)C)ccc(C#N)c(NC2CCN(C(=O)CCc3nnc(C)n3C)CC2C)n1 C1(C(=O)NCC2CCCN2C(c2cc(Cl)no2)=O)CCC(=C2CCC2)CC1 c1(C(N2C(C(=O)NC(CC(C)(C)C)CO)CNC(=O)C2)=O)cc2ccccn2c1 CC(C(=O)N(C)CC1(NC(=O)CC2CC2(C)C)CC1)c1cc[nH]n1 C1(OCC)CN(c2nnc(CC(C)O)n2CCOC)C(C)(CC)C1.C(C=O)OCC C(N=c1nc(N2CCN(C)C(CO)C2)c2sccc2[nH]1)C1CCN(C)C1 c1(CC)cc(Br)ccc1C(=O)Nc1cccnc1C(N1CCC(C(=O)OC)C1)=O CC(C)C(C)(O)C(=O)N(CCOCCNC(c1ccc(CN(C)C)cc1)=O)C c1(C(N2CC(CNC(C3(C(=O)NC)CCC3)=O)(OC)C2)=O)c(C)cc(C)nc1O CC(C)CC(C)CC(=O)NCC1CCC(C(N2CC3OCC(CO)C3C2)=O)C1 Cc1c(C(N2CCC(NC(C3CCc4nn[nH]c4C3)=O)C2)=O)c(O)ccc1F c1(CNC(C)=O)ccc(C(=O)NC2CC2SCCS(C)(=O)=O)o1 O=C1CCN(C(c2ccc(Cl)o2)=O)C2CCN(C(=O)Cc3cscn3)CC2N1 c1(C(=O)NCCNC(c2cccc(C)c2F)=O)c(C2CC2)nc2sccn12 C(CC(=O)NCC1CN(C(C2(C)CC=CC2)=O)C1)(C1=CCCC1)OCC CC1=C(C(=O)NCC(N2CCN(C(=O)C3=CCCC3)CC2)=O)CCO1 N1(C(c2ccc(Br)cn2)C(=O)NCc2ccc(F)cc2)CC2CCCC12 C1(CN(C(C(=O)NCCCC)c2cccs2)C)CCCC12CC2 Cc1ccc(C(N2CCOCC(CNC(=O)COc3ccsn3)C2)=O)cc1C C1(C(C)(C)O)CN(C(C2CCN(C(=O)NC3(n4ccnc4)CC3)CC2)=O)CCO1 C1(C(C#C)C)CCN(C(=O)C(CNC(=O)Cc2csc(C)c2)C2CC2)CC1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC2(CCN(C(CCCOC)=O)C2)C1 N1(C(C(C)(C)F)=O)CCC2(CC1)CC(NC(=O)CCN1CCCC1=O)C2 CN1CCN(C(=O)C=C2CCCCC2)C(C(N2CCC=C(F)C2)=O)C1 Cc1c(CC(N2CCC(NC(C3CC(=C4CCC4)C3)=O)C2)=O)cccc1Br c1(C(=O)NCC2C(NC(C(C)Cc3ccco3)=O)C2)cc2ccsc2c(O)n1 c1(C(=O)NC2(C)CN(C(c3c(CCC)n(C)nc3)=O)C2)cc(F)ccc1OC C1(N(C(CC2C(CC)C2)=O)C)CN(C(=O)CCC2CCC(=O)N2)CCC1C N1(C(c2scc(C(N)=O)c2)=O)CCC(NC(c2ccsn2)=O)C1c1ccccc1 N1(C(C(CCSC)OC)=O)CC(NC(c2nnc(C)s2)=O)CC12CCCCC2 Cc1ccc(OCCC(=O)NC2(CNC(c3cnccc3Br)=O)CCOC2)cc1 C1(NC(C2C(C(=O)OCC)C2)=O)CC(C)CN(C(c2cc(OC)n(C)n2)=O)C1 C#CCCCCCCC(=O)NCC(C)N(C(=O)C(C)=CC1CC1)C C(=O)(C(C(=O)N(CCCNC(c1ccc(C)nn1)=O)Cc1ccccc1)OC)OC C1(C(=O)NC2CCCC(CC(=O)N(C(CSC)C)C)C2)CC2C(C1)C2(F)F c1(C(N(C2CN(C(=O)CSCc3ccc(F)cc3)C2)C)=O)cn(C)c(=O)nc1O Cc1cccc(COC(=O)C(=O)Nc2ccc(Br)cc2Cl)c1C C1(c2cn(CCC(=O)OC)nn2)N(C(=O)CC2CC(=O)NC2=O)CC12CCC2 C(C(C)C(=O)NC(C)(C)CNC(C1(C2CCCO2)CC1)=O)SC c1(C(=O)NCCCCCNC(C2C(CC)CCC2)=O)cc(C)nn1C(F)F c1(OC)cc(Cl)c(Cl)cc1C(N1CC(NC(=O)C(O)Cn2cncn2)C(O)C1)=O Cc1nc(NC(c2cc(C3CCC3)on2)=O)cc(O)n1.c12cccc(c1)NC2=O C(=O)(CN1C(=O)Cc2ccccc21)NC(CN(C(c1cnccc1Cl)=O)CC)C CC(C)(C)C(C#N)C(=O)N1CCCCC1CNC(c1ccc(-c2cc[nH]n2)s1)=O c1(C(N2CC(NC(=O)CC3COCC4(CCC4)O3)C2)=O)cc2cc(Cl)ccc2s1 c1(C(=O)NC2CC(CNC(=O)C(O)Cn3cncn3)C2)[nH]c2ccccc2c1Cl C(C(=O)NNC(=O)C(F)(F)CCn1ccnn1)c1n(C)c(=O)n(C)c(=O)c1C#N C1(N=c2nc[nH]s2)(C(=O)OC)CCN(C(=O)C2CSc3ccccc32)CC1 N1(C(c2ccccc2SC)C(=O)NC(CC)(C)C)CCC2CCOCC2C1 C1(C(=O)NCC(C)N(C)C)CC(O)CCN1C(c1cc(F)ccc1O)=O Nc1cc(C(=O)NC2CCCC(NC(=O)Cn3cc(CO)nn3)C2)c(F)cc1F C1(SC(C)(C)C)CC(NC(C2CCC2CNC(C2(CC3CC3)CCC2)=O)=O)C(O)C1 C1(O)(C(C(=O)NCC(CSC)OC)F)CN(C(=O)CCN(C)CCO)C1 c1(CC)[nH]nc(C(N2CC3C(C2)N3Cc2cccc(C(F)(F)F)c2)=O)c1F c1(CCNC(C2CC3CC3N2C(c2cocn2)=O)=O)ncccc1F C1(C(N2C(CNC(=O)CC3CCCOC3)CC(OC)C2)=O)CC(C(C)C)=NO1 CC(C)C(C(=O)NCCCN(C(=O)C=CBr)CCO)NC(c1ccccc1)=O Cc1c(C(=O)NC2CC2CNC(=O)CC2(C#N)CC2)cc(C2CC2)n1C c1(OC)ccc(OCC(=O)NCCNC(=O)CCCCOC)cc1 CCCCC(CC)C(=O)NC(C1(CNC(=O)CCSc2ccccn2)CC1)C C1(C(N(C)CC2CCN(C(CSCC#C)=O)CC2)=O)CC2CCCC2C1 c1(C(=O)NCC2(CO)CCN(C(=O)C3=CCCCO3)CC2)ccc2c(c1)CCO2 CC(C)(C)CCC(C)OC(=O)CCCCCC#N C(=O)(CCCCN=[N+]=[N-])NC(CCCC)C(=O)NCCc1nccs1 O=C(C1COc2ccccc21)NC1CCN(C(c2cccnc2)=O)C12CCC2 C1(C(N2C(C(=O)NCC34CCCCCC3C4)CC(=O)C2)=O)CCCC12CCC2 CCC(CNC(C1CC(O)C1(C)C)=O)(CC)NC(=O)C(C)(C)Oc1ccccc1 N1(C(c2ncc(CC)s2)=O)CCCC(C)(CNC(=O)C(C)(COC)OC)C1 N1(C(c2ncc(C)cc2C)=O)CCC2(CC1)CCN(C(C1CCSC(C)C1)=O)C2 Cc1cc(C)c(C2CCCN2C(=O)C(=O)N2CC(CC(C)N)C2)c(C)c1 C=CCCCCNC(=O)CCc1nnc(CN2CC(O)C2)s1.C(C)(C)(C)OC(=O)CO c1(CC(=O)NC(CC=C)Cc2ccccc2)cccc(CC2CC2)c1 c1(C(CC(=O)N(C2CCCC2C)CC2CC2)N(C(C)=O)C)ccc(F)cc1 N1(C(C2C(C)OCCC2)=O)CC=C(CCNC(c2cn(C)c(=O)nc2O)=O)CC1 C1(C(=O)NC(c2cncnc2)C)CC2(CCN1C(=O)C(CO)N(C)C)CC2 c1(C(N2C(CNC(CCS(C)(=O)=O)=O)CC2)=O)cc2c(nc1O)CCC(F)(F)C2 C(=O)(C1c2ccccc2CN1S(=O)(=O)CCCOC)N(CC(C(=O)NC)C)C c1(CC(=O)NCC2(NC(C=C(C)Cl)=O)CC2)cc(C)cc(C)c1 N1(c2nc(=N)nc(N3CCCCC(CC)C3)[nH]2)CCCC2(C1)OCc1ccccc12 N1(C(Cc2ncc(CC)s2)=O)CCCC(NC(C2CCCCN2CC)=O)C1 Cc1cccc(C(C)N(S(=O)(=O)CC2(CC(=O)O)CCCCC2)C)c1 C1(C(=O)NCCOC2CCN(C(CSC)=O)C2)NC(=O)C2CCC12 Cc1[nH]c2ccc(C(N3CCN(C(=O)C=Cc4ccsc4)CC3)=O)cc2c1C C1(C(N2CCC(=CCNC(C3C(C=C)C3)=O)CC2)=O)CC2CCC(C1)C2F CN1CC(C(=O)NC2CCCC2NC(C2(c3ccnn3C)CC2)=O)NC1=O N1(C(c2nc(CCC)sc2)=O)CCN(C(=O)C=C(C)Cl)C(c2cccc(Cl)c2)C1 Cc1ccc(N)cc1C(N1CCC(CO)C(NC(=O)CCC2CCCC2)C1)=O C12CCCN1N1CCN(CC1C)CCC(=O)C2.CC1CCN(CCO)CC1 N1(C(CN(C(C)=O)C)=O)CCN(C(=O)CC2CC3(CCC3)CO2)CC(C)C1 C1(C(=O)NC)CCN(C(=O)C(C2CCN(C(C(=O)C(C)(C)C)=O)CC2)O)C1C C1(C(=O)NCCC2(NC(c3sccc3C)=O)CCCC2)(NC(C)=O)CCCCC1 c1(OC)ccc(C(C)C(=O)NC(C2CN(C(=O)Cn3nccn3)C2)C)cc1 C(=O)(CCCC1CCOCC1)N(C(C)C(=O)OC(C)(C)C)C C(CCN=C(NCCS(C)=O)NCc1ccc(CS(C)=O)cc1)SC C(CN=c1[nH]c2ccccc2s1)N(CCOC(C)C)C(C1CCCC(C)C1)=O N1(C(C(C(C)C)F)=O)CCN(C(=O)CNC(=O)C2CC2)C(CCO)C1 N1(C(c2c(C)cc(C)s2)=O)CC2CCC1C(NC(c1cc(S(N)(=O)=O)c[nH]1)=O)C2 C1(C(=O)NCCC(C)NC(C2(O)CC3(CCOCC3)C2)=O)CC(C)(C)C(C)(C)C1 C(=O)(C(C)CCOC)N(CCC(=O)NC(c1nccn1C)C)CC#C c1(C(=O)NCC23CN(C(C=CC(C)C)=O)C(C2)CO3)cnc2ccc(F)cn12 c1(C(N2C(CNC(=O)COC3CCCC3)CC(O)C2)=O)csc2c1CCCC2 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CN(C(C3CCCN3N=O)=O)CC2C1 Cc1cc(=NCC2CCN(C(c3cc4c([nH]3)CCC4)=O)CC2C)[nH]c(C)n1 C(=O)(C1CCCn2ncnc21)N1CCC(NC(=O)Cn2ncc3ncccc23)C1 c1(C(=O)OC)cc(Cl)n[nH]c1=NCCN1CCC(OC(F)F)CC1 c1(CCNC(C(C2CCCC2)NC(C)=O)=O)nccc(C)n1.C1(=O)C(C)O1 c1(CNC2CN(Cc3ccc(OC)nc3)CCCO2)ncc(C)c(OC)c1C C#CCC(CC#C)NC(=O)CC1CN(C(c2cccc(Cl)c2)=O)C1 CCCCCC(O)C(C)C(=O)NNc1cc(C(=O)OC)cc(F)c1 N1(C(C(=O)NCc2ccco2)c2nccs2)CCCCC1CCF N1(C(C(CC)C)=O)CC(C2CCN(C(=O)Cc3ccc(CC(C)C)cc3)CC2)C1 N1(C(c2c(C)cco2)=O)CC(NC(=O)C(C)(C)c2cc[nH]n2)C(N=[N+]=[N-])C1 C123CCCC1N(CC2)C3=O.C1(N(C)C)(C(=O)NCC2CC23CC3)CCCC1 C1(NC(c2c(C)nc(C)[nH]2)=O)CC2CCC(C1)N2C(C1CCCC(C#N)C1)=O C1(C(=O)NCC(CC)NC(=O)CCN2CCNC(=O)C2)CCCNS1(=O)=O CC(CC(=O)N(C12CCC(CC1)C2)C)C(C)(C)NC(c1cc2cc[nH]c2cn1)=O N1(C(=O)NCC2CCCO2)CCn2c(cnc2Cc2cccc(C(=O)OC)n2)C1 N1(C(c2cccc(C)c2Cl)=O)CC2=C(C1)CN(C(=O)C(N1CCCC(O)C1)C)C2 S(=O)(=O)(c1csc2ccccc12)N1CCN(C(=O)Cc2ccc(O)cn2)C2C1C2 C1(C(=O)NCCCN(CCCNC(=O)CNC(N)=O)CC)CN2CCCC1CC2 c1(CCC(=O)NCC2(CNC(C3COC(=O)C3)=O)CCOCC2)cccc(Cl)c1 C(C)(C(=O)NC1(CSC)CC1)(C(C)C)OC.C12CCCC(C1)CC(=O)N2 N1(C(=O)COC(F)F)CCN(CC23CCC(CC2)CC3)CC1CO c1(C(=O)NCC(CNC(C2C(CC)C2)=O)F)cc(Cl)c(Cl)cc1C c1(C(=O)NCC2C3CN(C(CC4CCC(=O)NC4)=O)C2C3)ccc([N+](=O)[O-])[nH]1 C1(C(F)(F)F)(C(=O)OC(C)(C)C)CC=CCO1.C12CCC(C1)C(=O)NC2 CCCC(CNC(=O)C(O)CCN(C)C)C(=O)NCC1(F)CN(C)C1 C1(NC(C(C)NC(=O)NC)=O)C2CCC1CN(C(=O)C(N)=O)C2 c1(COC)cc(=NC(=O)C(C)(C)C(C)(C)NC(=O)OC(C)(C)C)[nH]n1C C1(C)(C(N(CCC(C(C)C)NC(=O)C(C)S(C)(=O)=O)C)=O)CCCS1(=O)=O c1(CCC(=O)NC(C2CCCCC2)CNC(CCOC)=O)nc2cc(Cl)ccc2s1 C(C(CC(=O)NCCC(O)C(C)C)C1CC1)NC(C1C(CCOC)C1)=O C1(C(=O)NC2CC(NC(=O)CCOCC(F)(F)C(F)F)C2)CC2(C1)CC(O)C2 CC1CCN(C(=O)C)CC1.C1(C(C(=O)N2CCC2CN=[N+]=[N-])N)CC=CCC1 C1(O)(CCNC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)CCc2ccsc2)CC1 c1(C(C(=O)N(CC(O)CNC(=O)CSCC2CCCO2)C)(F)F)ccc(F)cn1 C(CC(C)C)(C(=O)NCc1cn(CC)nc1C)NC(CSCCC)=O n1(C(C(N2C(CCNC(c3c(C)csc3)=O)CCC2)=O)C)c(C)cc(O)cc1=O C1(CCC)CN(C(=O)CNc2ccccn2)CCN1C(=O)CC1(CO)CCC1 N1(C(C(CC)(C)O)=O)CC(CNC(=O)C=Cc2ccnn2C)OC2(CCC2)C1 CN1CCCC(O)(CC(=O)NCC(C(C)(C)C)NC(c2ccncc2O)=O)C1 Cc1cnc(C(N2CC(NC(C3CCSC(C)C3)=O)C(C)C2)=O)cn1 CCC(C)(C)C(O)C(=O)N1CC(CCNC(=O)C(C(C)OC)N(C)C)C2(CC2)C1 C(=O)(CC(C)CC(=O)OC)NCCN(C(=O)CCc1cccnc1Cl)CC C1(CNC(C(C)O)=O)C2CCCC1N(C1=Cc3nncn3C1)C2 N1(C(CC(C)CF)=O)CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1C1CC1 Cc1ccc2[nH]c3c(c2c1)CC(C(N1CCOCCC1C)=O)CC3 N1(C(c2c(C)cno2)=O)CCC2(CC1)CC2NC(c1nc(Cl)c(Cl)s1)=O C(CC(C)(C)CC(=O)N1CCC(CCC(=O)NC2COC3(CCC3)C2)CC1)OC C1(C(=O)NC2C(C)N(C(C3CC3Cl)=O)CCC2)CCC2(CCCC2)C1 CN1CC(=O)N(CC(=O)NC(C)(C)CCCNC(C2CCC(O)C2)=O)C1=O c1(C(C)(C)C)cc(C(=O)NCCOC2CCN(C(C3(C#N)CCC3)=O)C2)on1 CCCCCCC(=O)NC1CCN(C(=O)CN2CCC(N(C)C)CC2)C1 N1(C(CC2CC(CN(C)C)C2)=O)CCN(C(c2cncn2C)=O)CC1 C1(F)(SCNC(C2CCCCC2)=O)CCCN(C(=O)COC2CC=CC2)C1 c1(C(=O)NCC2CN(Cc3c(CC)nns3)C2)cnnc(-c2ccccc2)c1 N1(C(C=Cc2cn(C)nn2)=O)CCC2(CCC2NC(C2COCCO2)=O)CC1 c1(NC(C(CO)N(C)C)=O)ccc(CNC(=O)CSCc2ccccn2)cc1 C1(C(=O)NCCCCNC(c2ccn(C)c(=O)c2)=O)CCCCC(F)(F)C1 C1(CNC(C2C(NC(C3(COCC)CCCC3)=O)C2)=O)(CO)CCSCC1 CC(c1ccco1)=CC(N1CCOC(CCNC(=O)CCc2ccc[nH]2)C1)=O Cc1ccc(NC(=O)C(C(C)(C)C)c2ccccc2)c2nsnc12 N1(C(CCC(=O)OC)=O)CC(NC(c2ncc(Br)cc2C)=O)C(C#N)C1 c1(C(C)C(=O)NC2CC2c2ccccn2)cc(F)cc(F)c1 c1(CC)cc(N)c(C(=O)NC2CC2CNC(=O)Cc2cc(Cl)cc(Cl)c2)c(F)c1 C1(NC(=O)NC2CCN(Cc3ccccc3)C2)CCC12CCCC2 C(=O)(CC1=CCCCC1)NC1CC(CCNC(C2CCC(OC)CC2)=O)C1 C1(OC)CC(NC(=O)CCS(N)(=O)=O)CN(C(c2nc(C(C)C)ncc2Cl)=O)C1 c1(OCC(=O)NCC(N(C)C(C2CC3CC3C2)=O)C2CC2)ccc(F)cc1O N1(C(C=CC(CC)C)=O)CC2CC1C2NC(c1ccc(C2CCCCC2)o1)=O c1(COCC)cc2oc(Cl)cc2[nH]1.c12cc(nc(C(F)(F)F)n1)NC1CCN2C1 C12(CNC(C(C(C)C)O)=O)CN(C(C3CCOC3C)=O)CC(F)(C1)C2 C1(C#N)(CN(C(c2csnc2C)C(=O)NC2(C)CC2)CC)CCOCC1 CCC(C)(C(=O)NCC(C1CC1)N(C)C(c1n[nH]cc1Cl)=O)OC c1(CC(=O)N(C(CNC(CCC(=O)NCC)=O)C)C)ccc(OCC)c(F)c1 CC(C)CC(C)(C)C(=O)NC1CC(NC(C23CCCC(C(F)F)(CC2)C3)=O)C1 CN1CC(NC(=O)C(C2CCN(C(=O)Cc3cnoc3)C2)F)C2(CC2)C1=O N1(C(CNC(=O)OC)=O)CCN(C(C2CCC(=O)NC2)=O)CC1c1ncc[nH]1 c1(-c2ccc(CCC)s2)nc(CS(C)(=O)=O)nn1CCCCO N1(CCC)CCC(C(=O)NC2C3CN(C(c4n[nH]c(C)c4Cl)=O)CC23)CC1 CCCCCC(C)CC(=O)N1CCCC(O)(CNC(c2ccc(N)cc2F)=O)C1 N1(C(Cn2cc(C)c(O)nc2=O)=O)CCN(C(=O)CC2CC=CC2)C(C)CC1C c1(C2(C(N(CCCCCSC)C(C3CC3C(C)(C)C)=O)=O)CC2)cccc(C)c1.CO C(CC(C(=O)N1CCC(SC)C1)NC(=O)CCc1cnccn1)OC C(=O)(C(CC(C)CC)NC(=O)CC1CC(=C)C1)NC1C(C#C)CCC1 C1(C(=O)NC(CNC(c2cnc(CCCC)s2)=O)CO)CCc2nccn2C1 c1(CNC(C(CCOCC)NC(=O)CCc2ccccn2)=O)cc(C)cc(F)c1 CCC1CCC(NC(C2CC3CC3C2)=O)C1 C1(CC=C)(NC(=O)CCOC2COC2)CCCN(C(=O)C(C(C)C)OC)C1 C1(C(N(CC(CC)NC(C(C)=CCC)=O)C)=O)CCCCN1S(=O)(=O)CCCC C(=O)(CCCC(C)(C)C)NCCC(CC)(CC)NC(=O)Cn1ccc(Br)n1 C(=O)(CC(CNC(c1cc(C)sc1C)=O)C1CCC1)N(C(C(CC)C)C)C1CC1 c1(C(=O)NC2CCC(CNC(C=CCOC)=O)CC2)cc(N)c2ncccc2c1 N1(C(CCc2cc(C)on2)=O)CC2CCC1CN2C(c1coc(C2CCC2)n1)=O c1(CC)[nH]c(=N)sc1C(N1CC(CNC(=O)CCc2cncc(C)c2)C1)=O c1(C(N2C(CNC(C(C)C)=O)COCC2)=O)ccc2c(O)nc(O)nc2c1 C1(OC)CC(C(=O)N(CC(N2CCCC2)C)C)N(C(=O)CCc2ccn(C)c2)C1 Cc1cc(C)c2c(c1)CCC(C(=O)NC1CCC1NC(=O)CCC(C)(C)C)O2 N1(C(C#C)=O)CC2CC1CC2NC(c1ccc2c(c1)CC2)=O N1(C(CC=CC=C)=O)Cc2ccccc2CC1CNC(C1OCCC1C)=O N1(C(CC2(C)CC2)=O)CC2(CCN(C(c3ccc(CCC(N)=O)s3)=O)C2)C1 C#Cc1cc(C(=O)NC2CN(C(=O)CCCn3cncn3)CCC2F)cc(N)c1 C=CCC(Cc1ccccc1)C(=O)N1CC2CC2(CNC(c2cn(C)cn2)=O)C1 c1(CNC(CNC(C(C2CC2)OC)OC)=O)ccn(C)n1 CCC(C)CC(CO)NC(=O)C(c1ccccc1)NC(=O)C=CC1CCCCC1 C1(C(=O)NCCC(C(C)C)NC(=O)C(O)P(C)(C)=O)CCS(=O)(=O)C1(C)C Cc1cc(C#N)cnc1C(=O)NC1(C(=O)NC(CF)C(F)(F)F)CC(F)C1 c1(CC)nc(N2CCC(CN3CC(c4cc(N(C)C)on4)C3)CC2)cc(N)n1 Cc1c(Cl)sc(Cl)c1C(=O)NC(C)CN(C)C(C1CC1c1nccn1C)=O CCN=c1[nH]cc(C(N2CC(NC(C3(C)CCCO3)=O)CC2C)=O)s1 C12(NC(=O)CNc3ccc(F)cn3)CCC(CNC(=O)C=C3CCC3)(C1)OC2 c1(C(=O)NCCC2(CNC(c3nc(OCC)oc3)=O)CC2)ccc([N+](=O)[O-])s1 C(C(CNC(C1CC12CCCCC2)=O)S(C)(=O)=O)NC(C(C(C)C)F)=O CCC(CC)(CCNC(c1nc(C)ccc1F)=O)NC(c1cnc(C2CC2)[nH]1)=O C1(CNC(C2OCCN(C)C2)=O)C(C2CC2)CCN1C(C1CCCCC1(C)C)=O C1(CCC)CN(C(=O)Cc2cnc[nH]2)CC1NC(=O)CC1(O)CCOC1 C1(CNC(C(n2cccn2)OC)=O)CC2(CO1)CN(C(=O)Cn1cccn1)C2 CC(C)CCC(=O)C(=O)NC(CCC1CC1)C(=O)N(CCC(O)CO)C c1(CNC(C(C)OC2CCCC2)=O)cc(C(=O)N(C)CCO)no1 C(=O)(CCCC1CCC1)NC(C1CCCC1)CNC(C(C1CCC1)OCC)=O C12C3CC4C1C4C3C(=O)N2.N1(C(=O)OC(C)(C)C)CC(c2ccon2)C1.OC c1(C(=O)NC(CC=C)CNC(C2(C)CC2)=O)ccc2c(c1)nc(C)c(=O)n2C N1(C(C(C)SC(C)C)=O)CCN(C(=O)CCC2CCOC2)CC(O)C1 N1(C(C2(CC)CCC(C)(C)C2)=O)CCN(C(C2CCCC2OC)=O)CC12CCC2 c1(OC)c(CC(=O)NC2C3CN(Cc4cccc(Cl)c4)CC23)cccc1F c1(N2CCC(N3C(=O)OCC3)C2)[nH]c(=NCCC(F)F)nc2scnc12 c1(CC(=O)NCC2CN(C(CSCC)=O)C3C2C3)ccc(Cl)c([N+](=O)[O-])c1 C12(NC(CN(CCOC)C)=O)CC(CNC(C)=O)(C1)OC2C C(CCC(C)C)(c1ccccc1)Cc1ncc(CC)o1.C(=O)(C(=O)N)N C1(OCCOC)CC(N=c2[nH]c(=NCCC#CBr)[nH]c3cccnc23)C1 c1(C(=O)NCCCOCCNC(C(C)n2cncn2)=O)c[nH]c2c(Cl)cccc12 N1(C(c2ccc(C#N)cn2)=O)CC2CC(NC(C3(N4CCCC4)CC3)=O)CC2C1 C1(NC(c2c(C)nn(C)c2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CCC1CO Cc1nc(Cl)cc(Cl)c1C(=O)NC1CCCN(C(=O)COC(F)(F)F)C1 c1(NC(c2c(-c3ccc(C)nc3)nccc2)=O)ccc(Cl)c(C)c1 c1(C(N2C(C3(C(=O)NCC4(C(=O)OC)CC4)CC3)CCC2)=O)ccc(C#N)o1 c1(N(C(c2ccc(C)[nH]2)C(=O)Nc2ccc(Cl)cc2F)C)cccc(C)c1F C(=O)(CCCCCSC)N1CC(CN(C(C2N(C(=O)NC)CCC2)=O)C)OCC1 c1(CN(C(=O)C(SC)SC)CCO)ccco1.C(=O)(C=C1CCC1)CC#C C1(NC2CCN(c3nnccc3)C2)CC2(CCOCC2)O1 c1(C(=O)NCCCNC(C2CCC(C(=O)OC)C2)=O)c(C)oc(C)c1Br C12(NC(C=C(C)C(C)C)=O)CCC1CN(C(=O)Cn1ncc(Cl)c1C)C2 C1(NC(=O)NC(c2ccccn2)CC)CCN(C)CC1c1cnn(C)c1 N1(C(C(C2CCOC2)OCC)=O)CCC2CCN(c3cc(Cl)nc(C)n3)CC2C1 N1(C(CNC(N)=O)=O)CC2CC2C1CNC(C1CCCN1c1ncccn1)=O C1(C(C)C)(C(=O)N(CC(O)C2CC2)C)CCN(C(C2COCC2C(N)=O)=O)C1 c1(CC(N2CC3C(C(=O)NCCC(=O)N(C)C)(C3)C2)=O)ccc2ccccc2c1 c1(OC)ccc2oc(C(=O)NC3CC3CNC(=O)C(CC(C)C)OC)c(C)c2c1 N1(C(c2c(C)nn(C(C)C)c2)=O)CC(NC(=O)C(C)(C)CF)CC(O)C1 C1(CCC#C)CCCN(C(c2oc(CNC(C3(C)C=CCC3)=O)cc2C)=O)C1 Cc1cnn(C)c1C(=O)NCC(C)(F)CNC(=O)CCC(=O)C1CC1 C12(C(N3CC(C)C(NC(=O)CN4CSCCSC4)CC3)=O)CCC(F)(CC1)CC2 S(=O)(=O)(C(C)c1ccccc1)NC(C)COC1CCOCC1 C12(NC(C3C(C(C)C)CCC3)=O)CCC(NC(=O)COC3CC=CC3)(CC1)C2 C(=O)(C1=NNC(=O)C1)NCC1C(NC(Cc2cccc(COC)c2)=O)CCC1 C1(CC)(CC)CC(NC(c2cccc(O)n2)=O)CN1C(c1cnc[nH]1)=O CC(C)C(O)(C(=O)N1CCC1NC(=O)CN1C(=O)NC(C)(C)C1=O)C(F)(F)F C1(NC(COC(C)C)=O)CC(C2CCN(C(c3ccc(N)c(F)c3)=O)C2)C1 C1(C(C)NC(C(C)COc2ccccc2)=O)CCN(C(=O)C=C2CCC2)CC1 C(C(C)C)(C(O)C(=O)N(C)CCN(C(c1occ(C)c1C)=O)C(C)C)OC c1(N(C)C)cnc(C(=O)OCCN(C(C)=O)CC(C(=O)OC(C)(C)C)(C)C)nc1 c1(C(N(CCNC(c2csc(C(F)F)c2)=O)CC)=O)ccc2cnn(C)c2c1 C#Cc1ccc(F)cc1C(=O)N(C1CCN(C(c2c[nH]nc2C)=O)C1)C O=C(CC(C(F)(F)F)NC(C1CCCSC1)=O)NC1(C2CC2)CCOCC1 c1(C(=O)OCCCOc2ccc(F)cc2F)ccc2ncsc2c1 C1(CC(=O)COC(C2(C#C)CC2)=O)CCN(C(=O)CN(C)C(c2cccs2)=O)C1 N1(C(C(=O)NCC)=O)CC2CN(C(=O)COc3ccc([N+](=O)[O-])cc3)CC2(C)C1 Cc1cc(C(N2CC(NC(c3c(O)cccc3F)=O)C(O)C2)=O)ncc1Br C=CCC(C)(CC)C(=O)N1CC2(CC(CC#N)C2)C1 Cn1ncc(C(=O)N(CCC(=O)NCC2(O)CCSC2)CCCO)n1 c1(CNc2cncc(C(=O)NC)c2)noc2c1COCC2 c1(C(=O)NC(CC)CNC(c2ccn(C)c2)=O)ccccc1OCC(N)=O C12(C(N3C(C)CN(C(c4nncs4)=O)CC3)=O)CCCCC1OCC2 C(=O)(C1=Cc2ccccc2OC1)N1C(CNC(c2c(C)c(F)ccc2)=O)C=CC1 CCCCCCCCc1cn(CC2CN(C(=O)C(C)S(C)(=O)=O)C(C)(C)C2)nn1 C1(NC(C(CC)CO)=O)CC2(CCCN(C(c3cc(C)n(C4CC4)n3)=O)C2)C1 N1(C(C(CCC)F)=O)CC(F)(F)CC1(C)CNC(=O)CCC1CCCN1C c1(CSCC(C)C)ccc(C(=O)NC2CCCC2NC(c2cnsc2)=O)o1 CC(CCCCCO)NC(C1CCCCC1CNC(C1OCCC1C(C)C)=O)=O C1(CC(=O)NCCN(CCCCCC)C(c2cnn[nH]2)=O)CCCC(C(F)(F)F)C1 C1(CC#C)(C(=O)N(C)CCOCCN(C)C(C2CC(C(F)F)C2)=O)CCCCO1 N1(C(C(CCC)CNC(c2ccc3cccnn23)=O)=O)CCc2n[nH]cc2C1 N1(C(c2ccn(C(CC)CC)n2)=O)CC2CCC(NC(=O)C=C(C)C)(C2)C1 c1(C(=O)NC2CC(C)(CNC(C(C)n3ccnc3)=O)C2)ccnc(C(=O)OC)c1 CC1CCCN(C(=O)CN2CCC(O)CC2)C1CNC(c1cnn(CCF)c1)=O C(C(C)(C(=O)NCCCC(=O)NCCC1(O)CCOC1)OC)OC C1(CCN(C)CC2(CCc3ccccc3)CC2)CCN(C(=O)COC2CC2)CC1 C12(NC(CCCCN(C)C)=O)CCCCCC1N(C(=O)Cc1ccsc1)CC2 c1(CC)c2[nH]c(C)c1NC2=O.c1(C(=O)OC)ccc(N2CCOCC2)nc1 Cc1cc(CN2CC3C(CNC(=O)Cc4c(F)cccc4Cl)C3C2)cc(C)c1O c1(CC(CN2CCC(N(CCN(C(CC)C)C)C)CC2)N)cccc(Br)c1 C(=O)(CS(=O)(=O)CC)NC.c1(COC)nc(OCc2cn(CC3NCC3)nn2)n[nH]1 c1(C(=O)NC2CC3(CN(C(C4CN(CC(C)C)C4)=O)C3)C2)ccc(N)c(Cl)c1O Cc1nc(O)nc(O)c1CC(=O)NC1CC(F)(F)CC1NC(C1CC=CCC1)=O CC(C)C(CC(=O)NC(C)C(CO)NC(=O)CS(N)(=O)=O)c1ccccc1 C1(C(=O)NCC(CC)(C)Cl)CN(C(c2cc(C#N)cs2)=O)CCN1C C1(OC)CC(C(=O)NNC(=O)COC)CN(C2CC2)C1 C1(CNC(C(C)NC=O)=O)CN(C(=O)CC2CC3C=CC2CC3)CCC1C C(=O)(C(CNC(=O)CC1CC=CC1)CC1CC1)NCc1nc(CC)sc1 C1(N)CC2CCC1N2C(=O)C=CCOc1ccccc1.C1(C=O)C2CC3C(C2)C13 O=C1CCN(C(c2ccn(-c3ccccc3)n2)=O)C(C(F)F)C1 C1(NC(c2c(C)cc(F)s2)=O)CCC2(CCN(C(C3(N=[N+]=[N-])CC3)=O)CC2)C1 C1(NC(COC)=O)CC12CC(NC(C1(CO)CCCCO1)=O)C2 Cc1ccc(C=CC(=O)N(C2CC(C#N)C2)CC(=O)NCC(O)(CO)CO)cc1 C(CNC(=O)CCc1cncs1)(C(=O)NCCCN1CCC1)N(C)C C1(CNC(C(C2CCOC2)OC)=O)CN(C(c2cccc(F)c2)=O)CC1C(F)(F)F N1(C(C(C=C)CC)=O)CCC(C)CC1C(=O)NCc1ccn(CCF)n1 c1(OCC(=O)NC2CCCC(NC(CCSCCOC)=O)C2)cc(F)cc(F)c1 C1(CC)CN(C(=O)CC)CCN1N1CCC(c2ccccc2C)C1 C1(CC#C)(C(=O)NC(C)(CC)CC)CCN(C(c2nccs2)=O)C1 C1(C(=O)NCCc2c(CNC(C(CC)F)=O)nco2)CC12CCCCCC2 C1(NC(c2c(C)nn(CCC)c2C)=O)CCN(Cc2cc(CF)on2)CC1(C)C C=CCC(CC=C)C(=O)N1CCC1(C)CC(=O)NC(c1ncc(C)[nH]1)C c1(C(=O)NCC(CNC(=O)COc2cccc(C)c2)OC)cc(F)cc(F)c1O C(C1CCOCC1)=CC(=O)NCC1CC(NC(=O)COc2cccnc2)C1 S(=O)(=O)(C=Cc1ccccc1)N1CCN(C(c2cc(CC)[nH]n2)=O)CC(O)C1 C1(CN(C(CC2(NC(CCOCCC)=O)CC2)=O)C)COCCO1 c1(C(N2CC3C(C(N4CC5(CN(C)C5)C4)=O)(C3)C2)=O)ccc2cc[nH]c2c1 c1(C(=O)NCC2C3CN(C(c4cccc(C#C)c4)=O)CC32)ccc(C)c(F)c1F c1(C(=O)NC2C(CN(C(C(C3CC3)OC)=O)C)CCC2)ccc2c(c1)CC2 CC1CN(C(=O)CN(C)CCO)CC(C)N(C(=O)CC2CCOC2)C1 c1(C(=O)NCCCOC(C2CC(OC)C2)=O)nn(C)c2ccc(F)cc12 CC(CCNC(C1CCCCN(C(=O)Cc2cnns2)C1)=O)C(C)(C)C Nc1ccc(C(=O)NCC(c2ccccc2)CNC(C2(O)CCCCC2)=O)nc1 N1(C(c2c(C(C)NC(=O)C=Cc3cncs3)noc2)=O)CCC(O)CC1C1CC1 N1(C(C2(CC#C)CCCCO2)=O)CCC(NC(=O)C(C)CCCC)CC1C c1(NC(c2c(C)nc(-c3ccc(I)c(F)c3)s2)=O)cccc(C#N)c1 c1(C(=O)NC2CC(CNC(c3ccoc3Cl)=O)C2)ccc2cnccc2c1 c1(OC)ccc2c(c1)CC(C(c1nnnn1C)Nc1ccc3nc(C)sc3c1)CC2 Cc1ccc(C(=O)NCC2CN(C(c3ccc(N)cc3F)=O)CCC2C)c(C)c1 c1(CC)cccc(C)c1C(=O)NC(CO)C(C)NC(c1c(Cl)cccc1Cl)=O C1(C(C)C)CCC(C)CC1C(=O)NCC(O)CN(C(=O)CNS(C)(=O)=O)C C=C=CCN=c1[nH]c2c(c(=NCC3(C)CCOCC3)[nH]1)CCCC2 C1(C(=O)OC)(NC(=O)C(N2CCN(c3cc(C)ccn3)CC2)=O)CC(O)C1(C)C C1(COC)CC2(CCCN2C(c2ccc(N(C(=O)NC)CCO)c(C)c2)=O)C1 C1(NC(Cc2onc(C)n2)=O)CCN(C(C2OCCCO2)=O)CC1C C1(F)(CNC(CN(C(C)=O)C)=O)CCN(C(=O)Cc2cscc2Br)C1 C1(F)(C(=O)NC2CN(C(C=C(C)c3ccco3)=O)CC2F)CC2(CCC2)C1 CCCC(C#N)C(=O)NCC1CC1C(N1CCC2CCC12)=O N(C(=NCCC(=O)NC1CC1)NCc1ccc(-c2ccc(Cl)cc2)cc1)C1C(C)C1 C1(C2CCC(=O)NC2)(NC2CC(C)(C)CN(C(=O)OC(C)(C)C)CC2)CCC1 c1(C(N2CCCCC2CC=C)C(=O)NCCC)ccc(OC)c(C)c1 c1(C2(C3CC3NSC(F)F)COC2)nnnn1CC1CC1 c1(OCCCC(=O)NCCCC(C)NC(C2(C)CC2(F)F)=O)ccccc1F C(=O)(C1=CCS(=O)(=O)C1)N1CC(CCNC(CCc2ccc(N)c(F)c2)=O)C1 c1(C(N2CCC(NC(C(C(C)C)n3cnnn3)=O)C2)=O)ccc2ncccn12 CCC(C)C(C)C(=O)NCCCOCCN(C(=O)Cn1ccnn1)C C1(NC(C(CCC)F)=O)CC(NC(c2ncnn2CC)=O)C12CCC2 c1(C(N2CC(NC(C3(OCC)CCSCC3)=O)C2)=O)ncn2c1CCC2 C1(CF)CCN(CCSC2CC3CC3C2)C1 C(=O)(C(C)(C)CC(F)(F)F)N1CCOCC(NC(CC2(OC)CCCC2)=O)C1 C12(NC(CC3CC(OCC)C3)=O)CCCC(NC(=O)CCc3cnc[nH]3)(C1)C2 C1(C)(C(=O)NCCCN(C(=O)Cc2csc(Cl)c2)C)CCNC(=O)C1 C1(CC(=O)NCC(CNC(C2(F)CC3(CCC3)C2)=O)CO)CC(=O)NC(=O)C1 N1(C(CC2N(C)CCC2)=O)CCC(CNC(=O)COCc2cccnc2)CC1 c1(OC)ccc(NC(C2CC3(C2)CN(C(=O)CCC2CCCCC2)C3)=O)c(Br)n1 N(C(=NCCCCN(CC(F)(F)F)C)NC1CCCC1)Cc1c(C)noc1C C=CCCCC(C)(C)C(=O)N1CCC(OC)CC1.C12CCN(C(=O)C1)C2=O c1(C(N(C2CCCN(C(CCNC(C)=O)=O)CC2)C)=O)cc(F)c2c(c1)CCC2 N1(c2snc(COC)n2)CCC2(CCC2)C(NC(C2CC(F)C2)=O)C1 C(C(CC(C)C)C(=O)NCCc1ncc[nH]1)NC(C(CCC)F)=O c1(C(=O)NCC2CC(OC)CN2C(C2COCCO2)=O)cn(C)c(=O)n1C N1(C(=O)Oc2ccc(F)cc2)CC2CCC(F)(F)C2C1 c1(C(=O)NC2CCN(C(C(COCC)C)=O)CC2)ccc2cncn2c1 c1(NC(C2(c3ccc(Cl)cc3)COC2)C)nccc(F)n1 C12(C(=O)NCC(C(=O)NC(c3cccnc3)CC)O)CC(C)(CCO1)C2 c1(C(=O)NC2C3OCC(NC(COCC#C)=O)(C3)C2)ccc2c(c1)C=CCC2 c1(C(=O)NC(CN(C(=O)CCOC)CC)C)nsnc1O CC(C)CC(O)C(=O)NC(C)(C)CCCCNC(=O)Cc1cn2ccsc2n1 CC1CC(NC(c2cnc(O)c(Cl)c2)=O)CN(C(c2ccco2)=O)C1 C1(CCNC(CCC#C)=O)CCN(C(=O)CSc2nc(-c3ccco3)no2)CC1 C(CC(=O)N1CCOCCC1C)(C(F)F)NC(CCSCC)=O C1(C(=O)NCC2CCCSC2)(NC(Cc2cc(C)on2)=O)CCCC1C CC(CC1CCOCC1)C(C(=O)NC1CCCC1)N(C)CC1CC(F)(F)C1 C1(C(=O)NCCN(C(=O)Cc2cccc(OC(F)F)c2)C)CCCN(C(N)=O)C1 C1(CN(C(C2(C)C(C)C2)=O)C)CCCN(C(=O)C(C)(C)CC2CCC2)C1 N1(C(=O)Nc2ccc(C)c(N3CCCS3(=O)=O)c2)CCOC2C1C2(F)F c1(C(=O)NCC2C(NC(=O)C=C(Cl)Cl)C2)cccn2cnnc12 N1(C(CC2CC(C)C2)=O)CCC2(CCC(NC(=O)C3=NOC(C)C3)C2)C1 CC1CC(NC(c2ncncc2Cl)=O)CN(C(c2cc(Br)cn2C)=O)C1 N1(C(C(CCC)OC)=O)C2CCC1CC(N(C)C(c1cn(C)c(O)n1)=O)C2 C1(CNC(c2c(C)n[nH]c2)=O)CCC(CNC(C2CCCCC2C)=O)CC1 N(C1CCc2cccnc21)C(C1C(C)(C)CCN(C(=O)C2=NOCC2)C1)=O C1(NC(C2CC(O)(CC#C)C2)=O)CN(C(c2ccc(F)o2)=O)CC(F)(F)C1 c1(C(N(C2CCCN(C(C3(C)CC4CCC3O4)=O)CC2)C)=O)ccc(F)cc1Cl C=CCC(CC(C)C)C(=O)N1CC2(CCC(NC(=O)C(O)C(F)F)CC2)C1 C(=O)(C#CC(C)(C)C)N(CCC(N1CCCCC1CN(CC(F)(F)F)C)=O)CC C12(C(=O)NCC(C)CNC(=O)CSC(F)F)CC3CC(C1)C(=O)C(C3)C2 c1(CCCSCC(=O)NC2C(NC(C3(C#N)CC3)=O)CC2)ccccc1 CC1COc2ccc(C(=O)NCCC(C)(C)CNC(c3cccs3)=O)cc21 CCC(O)C(C)C(=O)N1CCCC(C(C)(C)C(=O)NCCCc2ccncc2)C1 c1(C(=O)NC(C)CCNC(C2(C(N)=O)CCC2)=O)cc2c(Br)coc2cn1 CC1CCCC(C(=O)NC2CC(CNC(C3(CC(F)F)CCC3)=O)C2)CC1 N1(Cc2cc(OC)cc(Br)c2)CCC(NC(C2CCCCC2OC)=O)C(C)(C)C1 CCC(C)(C(=O)N1CCCC(NC(c2ccnn2CC#N)=O)C1)C(N)=O C=CCCC(C1CC1)NC(=O)COC1CC(CNC(=O)CC2CC2(C)C)C1 c1(CNCC2CN(C(=O)OC)C2)ccc(-n2cc(C)cn2)cc1 CCC(COC)C(=O)NCCCCNC(C1C(c2ccccc2)C1(F)F)=O N1(C(C2C(=C)C2)=O)CCC(O)(CN(C)C(c2oncc2CC)=O)C1.CC c1(C(C)C)ccc(-n2cnc(NCC(=O)CNC(=O)OC(C)(C)C)c2)cc1 c1(CC)cc(OC)ccc1C(=O)NCC1COCCN1C(=O)Cc1ccnn1C n1(CC)ncc(C(=O)NCC(C)N(C)C(C2(C)CC=CCC2)=O)c1Br c1(CC)ncc(CNC(=NC)NCC2CCOC2CCN2CCCC2)s1 C#Cc1cccc(C(=O)NC(C)CCCNC(=O)Cc2cn3ccsc3n2)c1F Cc1ccc(C(=O)NC(=O)C(C)NCc2ccnn2-c2cccnc2)cc1 N1(C(C(C)OCC)=O)CCN(C(=O)C(C(C)C)n2cncn2)CC(O)C1 C12(COC(=O)CSc3ccc(F)cc3)CC(CC1C(F)(F)F)C2 Cc1cc(CNC(C2(C)CCN(C(=O)CCC(C)(F)F)C2)=O)cnc1F c1(NC(C(CC)SC)=O)ccc(NC(C2CCC(C(N)=O)C2)=O)cc1.CCC#N N1(C(c2c(C)cno2)=O)CC2CC(NC(c3cnn(C)c3C(F)(F)F)=O)CC1C2 C1(C)(C(=O)NC(CN(C(CC2(CSC)CC2)=O)C)C)COCCO1 C(=O)(C1=C(C)OCC1)NCC1C(NC(C(CCC)c2ccc(Cl)cc2)=O)COC1 c1(OCC)cc(N2CC=CC(NC(=O)CC(c3cccc(F)c3)O)C2)nc(C)n1 C1(C(=O)NCC2CCC(C)C2)CN(C(c2ncccn2)=O)CC(C)O1 Cc1cc(C(=O)N(CCNC(C2CCC(C)S2)=O)C2CC2)c(N)c(Cl)c1 N1(C(CN2CCC(C)C2)=O)CC2CC2(C(=O)N(C2(C3CCC3)CC2)C2CC2)C1 c1(C(=O)NC(C(C)NC(C=CC(C)C)=O)(C)C)ccc(C#N)n1C CCCCCC(C)CC(=O)N1CCC(C(=O)NCCCC2(C)CC2)(OC)C1 N1(C(CCCC)=O)CCOC(CN2CCCC2CCNC(c2cnn(CF)c2)=O)C1 c1(N2CC(CN(C)C)OCC2)cc(Br)ccc1S(=O)(=O)N1CC2CCC2C1 c1(C(C)N(C)CC2(C3CCC3)CC2)ccc(Cl)cc1 N1(C(C)=O)CCOC(C(N2CCCC2C2(NC(C3CC=CCO3)=O)CC2)=O)C1 N1(C(C2C(C)OCCO2)=O)CCC(C(=O)NCCCC2(C)CC2)CC1C N1(C(C(c2ccc(F)cc2)C)=O)CC2CCN(C(c3cnc(Cl)[nH]3)=O)C2C1 Cc1cc(C(=O)NC2CN(C(=O)CO)CC2O)nn1C(C)C Cc1nc(C(N2CC(C)(NC(=O)CC3CC4CC4C3)C2)=O)cn1C C=CCN=C(NCc1ccoc1C)NCc1ccsc1C(=O)OC(C)(C)C C1(NC(=O)CCCc2ccncc2)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 c1(C(=O)NC(C)CNC(c2cc(-c3ccncc3)no2)=O)nnn(C)c1Br Cc1ccc(C(=O)N(C)CC2CN(c3ncnc(C(C)(C)C)n3)C2)cc1 c1(C(=O)NCC(CNC(C2CCC(C)CC2)=O)C)cccc2ncn(C)c12 O=C(C1=C(Cl)CCOC1)NCCC(O)CNC(C1(CC(F)F)CC1)=O c1(C(=O)NC(C)Cc2cn(CCCC(=O)O)nn2)nn(C)c2c1CCCC2 c1(CS(=O)(=O)NCC2(CS(C)(=O)=O)COC2)nc(Cl)cs1 C12CN(C)CCN1NC(=O)C1C23COC1C3.CC1CCCN(Cc2ccccc2)C1 Cc1occ(C(F)(F)F)c1C(c1nnnn1C1CCOC1)NC1COCC1F C(N=c1[nH]c(=NCC2OCc3ccccc32)[nH]c2c1CSC2)C1C(C)CCC1 CC(C)(CCCCNC(=O)COCc1ccccc1)C(=O)NNC(=O)CO C(C)(CCCCNC(c1ccc(C(C)(F)F)cn1)=O)NC(C(C)OCC(C)C)=O C(CC(O)CC(=O)N1CCOC(CCNC(=O)Cn2nnc(C)n2)C1)SC Cc1cc(NCc2cc(C3(C)CC3)on2)nc(=NCCCCN(C)C)[nH]1 C1(CNC(C2CC(=O)N(O)C2)=O)CC12CCN(C(=O)CCOCC1CCC1)CC2 c1(C(N2CC(NC(c3ccc(F)cc3Cl)=O)C3(C2)CC3)=O)cc(Br)ncc1Br C(C)(C(=O)NNC(=O)c1ccc(-c2cccc(CC)c2)o1)OCCCC C1(CNC(C2COCCO2)=O)CN(C(c2ccc(Cn3ccnc3)o2)=O)CCO1 C1(CCC)(NC(CC=C=C)=O)CCCN(C(c2cccc(C#N)c2)=O)C1 N1(C(C(C)(C)C#N)=O)CC2CCC(NC(=O)CC3(O)CCOC3)CC2C1 N1(C(CC(CC)C)=O)CCC(C(N2CCC(NC(=O)NC)CC2)=O)C(C)(C)C1 c1(C(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C2)ccc(F)c(C(F)F)c1 C=CCC(CCCCCC)C(=O)NC(C1CCN(C(=O)CN2CSCC2=O)C1)C NC(=O)CC(c1ccccc1)NC(c1cnc(C2CCCO2)s1)=O C1(CNC(C2CC3(CSC3)C2)=O)CCN(C(=O)Cn2ncccc2=O)CC1(F)F C(CCC(=O)N1CC(c2ccccc2)(NC(=O)CC2CCC(C)C2)C1)SC Cc1ncccc1C=CC(N1CC2(NC(C3CC(OC4CC4)C3)=O)CCC1C2)=O CC1CC2CN(C(c3nc(C4CC4)n4c3CCCC4)=O)CC2N1C(=O)C=CCO N1(C(C2CN(C)CC(C)O2)=O)C2CCC(C(=O)NC3(C)CCCC3(C)C)C1CC2 N1(C(CSCC#C)=O)CCC(F)(C(=O)NCCC2CCC(C)O2)CC1 Cc1cc(-c2ccc(C(=O)Nc3cnccn3)cc2F)cc(C)c1 C#CC1(C(=O)NC2CCCC2NC(=O)CCc2ccc(Cl)nc2)CCOCC1 CS(=O)c1cccc(NC(c2ncccc2C(F)(F)F)c2nnnn2C2CC2)c1 S(=O)(=O)(c1cccnc1)NC(C1CCCCS1)=O c1(C(=O)NCCCCN(C(CCN(CC(C(C)C)C)C)=O)C)occ2c1CCC2 Nc1cc(C(=O)NCC(CO)NC(=O)C(F)=CC2CC2)ccc1Br c1(C(N(C2CCN(C(=O)CCn3cc(Cl)cn3)CC2)C)=O)cc(C#N)ccn1 c1(OC)cc(F)c(C(N2CCC3(C2)CN(C(=O)CSC(C)(C)C)C3)=O)cc1OC C1(CNC23CC(C(=O)OC(=O)CS(=O)(=O)NC4CCCCC4)(C2)C3)CC12CCSCC2 C1(NC(C(CCOC)(C)C)=O)CCN(C(=O)C(C)(C)c2ccc(Cl)s2)CC(O)C1 c1(C(C(=O)NCCCCCC)N(C2CCCC2)C)sc([N+](=O)[O-])cc1Cl C12(C(N3C4C(NC(c5ccc6sccc6c5)=O)C(C4)C3)=O)CCCCC1OCC2 CCC(C)C(CC(=O)NCc1cc(OC)no1)NC(c1ccsc1Cl)=O c1(CC)nc(OC)cc(=NC2CCCC(SCC3(CSC4CC4)CC3)C2)[nH]1 c1(C(N2CC(C)(C)C(NC(=O)CCC(N)=O)CC2)=O)ccc2c(c1)COCC2 CCCC(C)(CC)C(=O)N1CCN(CC(C)NC(c2cc(C3CC3)ns2)=O)CC1 CC1(C)CCCC(C(=O)NC(C)(CNC(c2c[nH]nc2F)=O)CO)C1 c1(C(N2CC(C(C)Nc3ncc(O)cn3)OCC2)=O)ccnc(Cl)c1F c1(C(C(=O)NCC)N(C)CC2CC=CCC2)ccc(C=NOCC#N)o1 Cc1oc2ccccc2c1CC(N1CCN(C(=O)CC(F)(F)Br)CC1)=O Cc1nnc(CC(=O)NC2CC(C(=O)OCC3(F)CC(CO)C3)NC2)n1C c1(C(N(C(C)CNC(=O)CN2CCCC2CO)C)=O)cnn2cccc2c1 N1(C(C2(CC(N3CCC4C(N(C)C)C4C3)=O)CC2)=O)CC2(C1)CC(C)(F)C2 CCCC(C)(C)NC(=O)NCc1ccc(-c2cnn(C)c2)o1 Cc1nc(CC(=O)NC2CC(NC(=O)CN(S(C)(=O)=O)C)C2)c(C)s1 C=CC1(CO)CCN(C(C2COC(CNC(c3cccc(CC)n3)=O)C2)=O)CC1 c1(NC(N2CCN(C(=O)NC)CC2)=O)ccc(N(C)C)c(Cl)c1 c1(C(=O)NC(COC)CNC(c2cocn2)=O)cccc(N(C)C)c1 O=C1CCc2cc(S(=O)(=O)N3CCC(c4cc(C)[nH]n4)C3)c(Br)cc2N1 CCCC(CC)CCC(=O)N(CCC(C(C)(C)C)NC(C12CCC1CC2)=O)C C#Cc1cc(F)ccc1CN1CCC(C(=O)NCc2cncnc2)C1 C1(NC(C2(SC)CC2)=O)CCC(C)(CNC(=O)C(F)=CCCF)C1 C(=O)(CC(O)C(C)CC)N(C1(C(=O)NCc2ncc(CC)[nH]2)CC1)C c1(CC)ccc(C(N2CC(NC(=O)COC3CCOC3)CCC2C)=O)cc1F C1(C(N2CC(NC(C(C)CC3CCC3)=O)C(F)C2)=O)CCc2ccccc2CC1 c1(NC(c2n(CC)nnn2)c2cn(C3CCOC3)nn2)ccc(Cl)c(CO)c1 C1(C(N(C(CN(C(C2(CCOC)CC2)=O)C)C)C)=O)CCCC(O)C1 C=CCCC(CC(C)C)C(=O)N1C(CNC(C2(C)CCCO2)=O)CC2COCC12 C1(CC(C)NC(C2CC(C#N)C2)=O)CCN(C(=O)CCOC2CCCOC2)CC1 C1(CNC(COC(C)C)=O)C(CNC(c2cncnc2)=O)C1(F)F C#Cc1c[nH]nc1C(N1CCC1CC(=O)NCC1CC2(CC2)C1)=O C1(NC(C2C(C)OCCC2)=O)CN(C(C23CCCC(CO2)C3)=O)C2CCCCC12 c1(C(=O)NCC2C=CCN2C(c2cocn2)=O)ccc(OC(F)F)cc1Cl N1(C(c2c(C)nccn2)=O)CCC2(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)CCCC12 C(CCCC(c1nnnn1C1CCCCCC1)NC(C)(C)CCF)(OC)OC O=C(C1CCCc2ccnn21)N1CC2CC(C1)N(C(c1cncc(O)c1Cl)=O)C2 C12CCCN(C1)C(=O)C(C)S2.c1(C(N(C(=O)CO)CC)=O)ccco1 N(C(=NCCS(=O)(=O)c1cccs1)N1CC2C(CF)C2C1)Cc1nnc(CC)s1 N1(C(c2n(C)ncc2)=O)CC2CCN(C(C3COCCN3C=O)=O)CC2C1 CN1CCN(C(=O)CCCNC(C2CC2Cl)=O)CC1=O N1(C(c2c(COC)noc2)=O)CCC2(CCN(C(=O)C(C)(O)COC)CC2)C1 C1(NC(c2sccc2NS(C)(=O)=O)=O)CN(Cc2ccc(C)s2)CCC1CO C1(C(=O)NCC2C3CN(C(=O)C(F)C(F)(F)F)CC23)OCC2CCCC1C2 c1(C(=O)NCC2(C)OCCN(C(Cc3cn(C)nn3)=O)C2)onc2ccccc12 C(C(C)N=c1nc(OC)c2c([nH]1)CCCCC2)C1(CCCCCCCCC)CC1 n1(CC(N2CCCCC(NC(C(C)(O)C3CC3)=O)C2)=O)cnc2c(N)ncnc12 C1(CC=C(C)C)C(C)(C)CN(S(=O)(=O)CC2CC3(CCOCC3)CO2)C1(C)C N1(C(C(C2CC2)OCC)=O)CCC(F)(CNC(c2c(C)coc2CC)=O)CC1 C1(CC=C)(NC(CSCCCC)=O)CCCN(C(C2(C)CCNC2=O)=O)C1 CCC(C)(CNC(C1(C#N)CC(=O)C1)=O)CNC(c1coc(SC)c1)=O N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)CC(C)(O)COC)C(C)(C)C1 N1(C(CCC(=O)NCCC)=O)CC2(CCN(C(=O)C(O)CC)CC2)CC1C C1(NC(c2occ(C)c2)=O)CCCC12CN(C(c1cc(Cl)cc(Cl)n1)=O)C2 N1(C(Cn2c(C(C)C)ncc2)=O)CCC2(NC(=O)CCN3CCC3)CCCC12 c1(N(C2CCC2)CC2(Cl)CC2(F)F)ccc(S(=O)(=O)NC(=O)OC(C)(C)C)cc1Br N1(C(C2OCCC(C)(C)C2)=O)CCC(C(=O)NCCN(C2CCC2)C)CC1(C)C C1(C)(CNC(C(C)NC(C)=O)=O)CCCN(C(=O)CCS(N)(=O)=O)C1 C1(COC)(CO)CC1C(F)(F)F.C1CCNC(=O)N1 CCC(CC)C(F)C(=O)NCCn1cccc1C(=O)NC(CC)CCO N1(C(c2ccccn2)C)CC(C(=O)O)Nc2ccccc21 N1(C(c2c(C)ccs2)=O)CCN(C(C2Cc3ccc(F)cc3O2)=O)C2(CCC2)C1 C1(CNC(C2C(C)(C(C)C)C2)=O)CCCCN1C(=O)CCF C1(C(C(=O)NCC(C)(CSC)OC)O)CCCCCCC1 N1(C(C(C)OCC=C)=O)CC(C(=O)NCC2OC(=O)CC2(C)C)CC(C)C1 N1(C(c2sccc2CO)=O)CCC(OCC(=O)N(CCO)C2CC2)C1 C1(CNC(c2c(CC)scc2)=O)CN(C(=O)C(=O)N(C)C)CCO1 CCS(=O)CC(=O)N1CCC(C)C1CNC(=O)Cn1ccnn1 c1(NC(C(=O)NCc2cc(C3CCC3)no2)=O)ccc(S(=O)(=O)CC2CC2)cc1 C=CCCC(O)CN(C)C(c1sccc1CNC(=O)CC1CC1(C)C)=O Cc1ccc(-c2ncccc2C(N2CCOC(COC(F)(F)F)C2)=O)cc1OC C=C=C(C)CC(=O)NCCC1CCN(C(c2ccc(C3CC3)nn2)=O)C1 N1(C(C(C)Br)=O)CCCC2(CCCN2C(=O)C(C)Oc2ccccc2)C1 C=CC(CC)C(=O)NC1CCOC(CNC(=O)CCc2nccn2CC)C1 C(C(C)C(=O)NC(C)(C)C(C)NC(=O)CCc1ccsc1)OCC C(=O)(C1CCCc2cncn21)NC1(C2CCCN(C(C3(C(C)C)CC3)=O)C2)CC1 C(=O)(C(CCC(C)NS(=O)(=O)c1c(C)nn(CC)c1Cl)C(=O)OC)OCC Cc1cc(F)ccc1NC(C1(C)CCN(C(C2CC2C(C)C)=O)CC1)=O N1(C(C)=O)CC(O)CC1C(=O)NC1CC2C=CC1C2.c12ncc(o1)c(=O)[nH]2 Cc1cnn(C)c1C(=O)N(C(c1ccccc1)CNC(=O)CCS(C)=O)C c1(C(=O)NCCC(=C)CNC(=O)C=CC)ccc(-n2ccnc2CCCC)cc1 C1(C(N2C(C(C)(C)NC(c3cc(F)c[nH]3)=O)CCC2)=O)CCCCS1(=O)=O C1(C(=O)NCC(C2CCN(C(=O)C(F)(F)C3CC3)CC2)(C)C)CN2CC(=O)CC2C1 CCC(C)(C)CC(=O)N1CC(CN=c2[nH]nc(C(N)=O)s2)CC1C c1(CN2C(C(=O)NCCCNC(=O)C3CC3)CCC2)ccc(F)c(CO)c1 C1(C(F)(F)F)(NCC2(C(=O)OC)CC(=C)C2)CCc2ccccc2C1 c1(OC)ccc(C(N2CC(CNC(=O)Cc3ncc(C(C)C)[nH]3)C2)=O)cc1 N1(C(Cc2nn(C)c(Cl)c2)=O)CCN(C(C2(C)COCCO2)=O)CC1C1CC1 N1(C(C(CC2CC2)OC)=O)C(C(N2CCSCC2CO)=O)CCC1C1CC1 N1(C(C(CC)CC)=O)CC(C)CN(C(C2NC(=O)CC2C)=O)CC1C c1(C(C)NC)cccc(NC(c2ccnn2CC2CC2)c2nnnn2C)c1 c1(C(N2CC(NC(C(CCC)NC(N)=O)=O)C(CC)C2)=O)cc(C)nc(C)n1 c1(CC)cc(C(=O)NC2CC(N(C(=O)Cc3ccn(C)n3)C)C2)cc(Cl)c1 CC(C)(F)CCC(=O)N1CCC(CNC(c2cn(CC(F)(F)F)cn2)=O)CC1 N1(C(c2nc(Br)n[nH]2)=O)CCC(N2CCNCC2)C(F)C1 C(c1cnn(C)c1)=CC(N1CC(C(N)=O)(CNC(C2CC23CCOC3)=O)C1)=O N1(C(C=CCNC(=O)C=Cc2cc[nH]n2)=O)CCOC2CC12 N1(C(C2CCCN(S(N)(=O)=O)C2)=O)CCC2CCCC(C1)N2C(=O)C1=CCCC1 N1(C(C2CN(C)C2)=O)C2CCC1CC(N(C)C(c1ccc(O)cc1)=O)C2 C(=O)(C(C)CC(=O)NC(CCOC)C(=O)NC(C)C(=O)OC(C)C)OC C(CCCCC(=O)NC1C=CCCC1C(=O)NC1CCOC1C1CC1)N(C)C C(=O)(C(CNC(C1C2CCCCC12)=O)CC(C)C)NCCc1ncc(C)o1 C(=O)(CS(=O)(=O)c1ncc[nH]1)N1C(C)C(O)CCC1.c12cn(nn1)C(C)CC2 C1(C)(C(=O)NC2CCC(N(C(c3c(OCC)scc3)=O)C)CC2)CCCCCC1 C(=O)(C1=CCSC1)NC(CC)(C)CNC(c1cc(-c2ccc(Cl)s2)on1)=O Cc1cnc(F)cc1C(=O)NC1CC(C(=O)Nc2cc(=O)n(C)cn2)C1 c1(C(C)C)ccc(C(N2CCC(C)C2CNC(=O)CC(F)F)=O)c(Cl)n1 N1(C(CNC(C(CC)C)=O)=O)CC2CC1C2NC(c1cscc1C)=O n1(C2(CNC(=O)NCC3OCCN(C(C)C)C3)CC2)cnc2ccccc12 Cc1cccc(S(=O)(=O)NC2(C)CCc3ccccc32)c1F Cc1cc(C(N2CC(NC(=O)CCOC(C)C)C(CO)C2)=O)nn1C(C)C CN1CCN(C(C2C3CCCCC23)=O)C(CNC(c2cnn(C)c2Cl)=O)C1 c1(NC(C2CC3CC3N2Cc2cc(Br)c(Br)s2)=O)c[nH]c2cnccc12 c1(C(N2CC3COCCC3(CO)C2)=O)nc2ccc(-c3ccc(F)cc3)cc2o1 c1(CC)ccc(CNC(=O)NCC2(O)CCCC2(C)C)c(OC)c1 c1(CNC(C(=O)NC(c2ccc(=O)oc2)C)=O)occ2c1CCOC2 N1(C(=O)OCC)CCC(C)(C)C1CO.C1(C(C)C)C(=O)N2CCC2C(=O)N1 C1(C(N2CCN(CC=C)CC2)=O)CCN(C(c2occc2C)=O)C(C)C1 C#Cc1cnc(C(=O)NCC(=O)NC2CC3CC3C2)c(C)c1 C1(N(C)C(C2CCCN(C(=O)C(=O)NCC(F)(F)F)C2)=O)CCOC(C)(C)C1 Cc1nccc(C(=O)NC(C(=O)NCCCc2ccccc2)c2ccco2)n1 c1(C(=O)NCCC2(OC)CN(C(CC=C)=O)C2)cc(C(C)=O)cn1C C(C(C)C(F)C(=O)NCc1noc(COC)n1)NC(CSCC(=O)OC)=O C(=O)(C1=NOC(C)C1C)N1CC(C(=O)NC(CC#C)CO)C(CCC)C1 N1(CCNC(c2coc(C(F)F)c2)=O)CCCN(C(C2CC2C2CC2)=O)CC1 C(C1=CCN(C(=O)C2=NOC(C)C2)CC1)NC(C(c1ccc(F)c(F)c1)C)=O N1(C(C)=O)CCC(C(=O)N(C)CCNC(c2sccc2CO)=O)CC1 N1(C(C2CCOCC2)C(=O)NCCCOC)Cc2cccc(C)c2C1 C1(C(=O)NCC(C)N(C(c2cnc(OCC)s2)=O)CC)CC2(C1)CC(C)(O)C2 c1(N)cccc(Cl)c1.C(=O)(C(C1CCSC1)N(CCN(C)C)CC)NCC N1(C2CC2)CSCC1C(=O)OCC.C(=O)(CC(=O)NCC)NC(C1(CNCC)CC1)C C1(C)(CNC(CCC(=C)C)=O)CN(C(c2nncn2CC)=O)C(C)(C)C1 C1(NC(C2=C(C)S(=O)(=O)CC2)=O)CN(C(C2COC(=O)N2)=O)C2(CCOCC2)C1 N1(C(c2c(CC)nccn2)=O)CCN(C(C2(O)CCC(CC)C2)=O)CC1C c1(C(N(CCN(C(C(F)=C(C)C)=O)C(C)C)C)=O)ccc(O)c(Cl)c1 C1(NC(C(C)OCC2CC2)=O)CCCN(C(c2cnc(Br)s2)=O)C1 c1(C(=O)NCC(C)(C2CC2)NC(C2CCc3cnnn3C2)=O)cnc2sccc2c1 N1(c2nc(SC)c(Br)cn2)CCC2(CC1)CC2C(=O)NC(C)CN1CCCC1 c1(C(=O)NCCN(C(C2COCC(C)O2)=O)CC2CC2)cc([N+](=O)[O-])sn1 N1(C(CCC2CCC(=O)N2)=O)CC2CCC1CN2C(C1CCS(=O)(=O)C1)=O C1(O)(CNC(c2c(CC)cncc2)=O)CCN(C(=O)CSCC(N)=O)CC1 N1(C(c2cc(I)nn2C)C(=O)NCCCCCC)CCOC(F)(F)CC1 C(C(=O)N1CC=CCO1)N(C(=O)CCc1cnccn1)C C1(CC(=O)NC(C)C(CO)NC(=O)CC2(O)CCCC2)COC(C)(C)C1 C(=O)(CCCC(C)(C)C#N)N(C(CC)CC(=O)NCC1CC1)C N1(C(c2c(OC)nsc2)=O)CC2CCC(C1)N2C(C1(C)CCC2CC2C1)=O N1(C(c2cc(SC)oc2)=O)CCN(C(c2nc(O)nc(O)c2N)=O)C(C)CC1C Cc1ccc(NC(C2CC2C2CN(C(C3CCCCC3)=O)C2)=O)cc1C#N C1(OC)CC2CCC1CC2C(=O)NC1COCC1NC(C1CCC(F)CC1)=O CCCC(CC1CCCC1)C(=O)N1CCC(CO)(NC(=O)Cc2ccoc2)CC1 CCC(C)CCC(=O)NCC1CC(C)CCN1C(=O)CSCCN(C)C N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC2CNC(c1cc(C)nc(C2CC2)n1)=O S(=O)(=O)(c1ccc(N2CCCC(N(C)C3CC3)C2)c(F)c1)N(CCOC)C Cc1ccc(C(=O)N(CC(O)CN(C(=O)CCC2CCCCO2)C)C)cc1CO C1(C(=O)NC(C)CCC2CCCCO2)CC(O)CN1C(=O)OC(C)(C)C N1(C(CNC(=O)OCC)=O)CC2CC1C2C(N1CC(N2CCC2)C1)=O C1(C(C(C)C)NC(c2nocc2Cl)=O)CCN(C(C2C(C#N)C2(C)C)=O)CC1 c1(-c2cnc(CC(=O)NCC3CCSCC3)nc2)ccc2c(c1)CCC2=O Cc1nnn(C)c1C(=O)NCC1(O)CN(C(C2CCC=CCC2)=O)C1 CC(C)C(C(C)NC(=O)CC(F)(F)Cl)NC(c1cncc(F)c1)=O CC(C)C(C)C(C)CC(=O)N1CCC(NC(C2Cc3nccnc3C2)=O)C1C N1(C(c2cnc(OCC)nc2)=O)CC2(CC2)CC1C(=O)NCCCC1CC1 Cn1nc(C(=O)NCC2COCC2NC(C2(C)COCCO2)=O)cc1C(F)(F)F N1(C(C2(CC)N(C(CC3ON=C(CC)C3)=O)CCC2)=O)CCC2(CC(CO)C2)C1 CN1CCOC(C(=O)NC2CCCC2CNC(=O)CCC2CCC(O)CC2)C1=O Cc1nn(CC(=O)NC(C)(CNC(=O)C=Cc2cn[nH]c2)C(C)C)c(=O)o1 C1(C)(C(=O)NCc2cc(C(=O)NC3C(OC)CCC3)n(C)n2)CCC(=O)NC1 C(=O)(CC(C)CC(C)C)NC1C(CC(=O)N(C(C(=O)OC)C)C2CC2)CCC1 c1(C(=O)NCC(CC)(C)NC(C2CN3CCCC3CO2)=O)cnc2[nH]cncc1-2 C(c1ccccc1C)=CC(=O)NCC=CC(=O)N(C)Cc1cnc(C)s1 N1(C(C2CCN(C)CC2)C(=O)NCC2CCCO2)CCOc2ccc(Cl)cc21 CC(CN(C)C)CCC(=O)N1C2CCC1C(CNC(c1cc([N+](=O)[O-])n[nH]1)=O)C2 c1(N2CCC(NC(CCSC)=O)C(C)C2)nc2cc(Br)ccc2o1 Cc1c(Cl)ccc(C(N2CC(CNC(c3ccc(C#N)cn3)=O)C(C)C2)=O)c1Cl O=C(C1=C(Cl)CCCC1)NC1CCC(O)CN(C(C2CCC(CO)CC2)=O)C1 CC1CN(C(c2cncc(C(N)=O)c2)=O)CC1NC(=O)CC1CCC(=O)N1 C(N=c1[nH]c(=NCCCC(=O)N(C)C)c2sccc2[nH]1)C1(CC)CCOC1 CC1CCN(C(c2csc(Cl)n2)=O)C1C(=O)NCC1(CO)CC(C)C1 c1(C(N2CC3C(CNC(c4n(CC)nnc4)=O)C3C2)=O)cncc2ncn(C)c12 N1(C(=O)Cn2ccnn2)CC2(C=C(C(=O)N3CC4C=CCC(C4)C3)CO2)C1 C1(NC(C(CCOC)NC(=O)C(C)=CC(C)(C)C)=O)CC2CCC1CC2 c1(C(N2CC(CNC(CCOCCC)=O)C(C)CC2)=O)cc2n(n1)CCOC2 N1(C(CCCn2cc(-c3cc(OC)nn3C)nn2)=O)CCCC(C)S(=O)CC1 c1(OC)ccc2c(c1)CCC2(O)CNS(=O)(=O)c1ccc2c(ccn2C)c1 Cc1cn2cc(CC(=O)NC3CC(NC(C4(CO)CCCO4)=O)C3)nc2s1 c1(C(=O)NC(C)CC2CN(C(C3CCC3(C)C)=O)C2)ccc(F)c2cnccc12 CC(O)CCCCCC(=O)NC1CC2CCC1N2C(c1ccccn1)=O C(=O)(C1CCOc2ccc(Cl)cc21)NCC1(C)OCCN(c2cc(C)ncn2)C1 C1(C)(CNC(CCSCC)=O)CN(C(c2ccc(C(=O)OC)o2)=O)C(C)(C)C1 CCCCC(CC)C(=O)N1CCC(CNC(c2nc(C)nn2C)=O)C12CC2 C1(CNC(c2cnccn2)=O)CCN(C(c2ccc3cc[nH]c3c2)=O)CC1(F)F n1(CCOC)nnnc1C(c1cnn(CC(C)C)c1)NC(C)(C)CSC c1(C(C)NC(=O)C(C2CC2)NC(C2CSC2)=O)cccc(O)c1 N1(c2cc(N3CC(CCO)OCC3)ncn2)CCCC2(CCNC2=O)C1 C1(NC(c2c(OC)n(C)nc2)=O)CCCN(C(c2cc(Br)oc2C)=O)CC1 N1(C(CCOC(CCC)=O)=O)CCN(C(C2CCC2OC)=O)CC1CC1CC1 C(=O)(CC1OCCc2sccc21)NCCCN(C)Cc1ccnc(Br)c1 C1(C(N(CCC(C)C)CC(=O)N(CCC)CCO)=O)CCN(C2COC2)C1 c1(C2NCCC(NCC(C)(C(F)F)OC)C2)c(C)cccc1Br C1(C(N2C(CCC(=O)NCC(C3CCC3)OC)CCC2)=O)CC(=O)N(C)C1 S(=O)(=O)(c1cccnc1Cl)N1CC2(CC(Nc3n(C(C)C)ncc3)C2)C1 N1(C(c2n(CC)ncc2)=O)CC(NC(=O)CNC(=O)CNC(C)=O)C2(CCC2)C1 C(=O)(CCCC(C)(C)C)NC1C(C(=O)NC(C)Cc2nc[nH]n2)C1(C)C N1(C(c2nc(CC)sc2N)=O)CCCC(F)(CNC(C2CC(CC)=NO2)=O)CC1 C1(NC(CC(=O)OC)=O)CC(CNC(=O)C(C)Oc2ccccc2CO)CC1O N1(CC(N2CCC(c3cccc(Cl)c3)C2)=O)CC(=O)CCC1=O.Cn1ccc(NC)n1 C12(CNC(c3cc(C)oc3)=O)CCC(C1)N(C(c1ncc(Br)cc1N)=O)C2 c1(C(=O)NC(C(C)(C)NC(CC(COC)(C)O)=O)C)ccc(CO)cc1F N1(C(c2c(OC)cccn2)C(=O)NC2CCOC2)CCc2c(Cl)cccc21 c12cc(ccn1)N2.CC1CCC(C(N2CCC2)=O)C1 C1(CC=C)(C(=O)NCCc2n[nH]c(C)n2)CCCN1C(=O)C(C)OCC c1(C(=O)NC(C(C)C)CCNC(C2CC(=O)N(C3CC3)C2)=O)ccc(O)c(O)c1 C1(OCCNC(C(C)n2ccnc2)=O)CCN(C(C2C(C(C)=O)C2(C)C)=O)C1 CC(C)C(CC(=O)NOCCC(C)C)NC(=O)C#CC(C)(C)C CCCN=c1nc(NCC(C)(C)C2=CCCCCC2)c2c([nH]1)c(C)nn2C C1(CNC(C2(Cl)CC2)=O)CCCN(C(=O)CC2=CCCC2)CC1 CC1(CCCNCC2CC(C(=O)NC3CC3)C2)CCC(=O)N1 C1(C2CC2)(COC)CN(C(c2conc2C(C)NC(=O)CC2CCC(C)O2)=O)C1 C1(Cc2n(N(C(=O)CC(C)(F)F)C(COC)=O)cnn2)CCS(=O)(=O)C1 C(=O)(C(C(C)C)NC(C1CCCN1Cc1ccc(OC(F)(F)F)cc1)=O)OC C1(=O)C(F)C(C)CN1.C(=O)(C(C)(C)NC(=O)C=CCCC(C)C)OCC c1(COC)ccc(C(=O)NCC2(F)CC(NC(C3CC3C)=O)C2)s1 N1(C(c2ccc(CC)cn2)=O)C(C(=O)N(C2CC(O)C2)C)CCC12CC2 N1(C(C2(CC)CN(C(=O)CNC(C3CC3C)=O)C2)=O)CCC(C(C)C)(CC)C1 N1(C(C(CC)=CC)=O)CCC2C(C1)CN2C(c1cc(OC)ccc1C)=O C(=O)(C(C#N)C(C)(C)C)NCCSc1cncc(C(=O)NCCCN(C)C)c1 C(=O)(C(F)(CNC(=O)C(C)=C1CCCC1)C(C)C)N(CCCN(C)C)CC c1(NC)ccc(C)cc1C(N1CC(O)(CN(C(=O)C(C)(C)CO)C)C1)=O C1(CC)C(C(=O)NCCCCN2CCCC2)CCN1C(=O)CC1CCCC2CC12 C1(OC)CCC(C(=O)NCCCCCN(C(=O)Cc2coc(C(F)F)n2)C)C1 CCCS(=O)(=O)C(C)C(=O)N1CC2CN(C(C3(C)CC(C#N)C3)=O)CC2(C)C1 CCC(C(=O)N1CCC(CNC(C2CN(CC(F)(F)F)C2)=O)C1)OCC C1(C(N2CC(C)(NC(=O)CC3CCC(O)C3)C2)=O)CCC2CC1CO2 N1(C(c2cccc(C#C)c2)=O)CCC2CCN(C(=O)C=C(C)C#N)CC2C1 n1(CC=C)cc(C(=O)NCC2CCCN2C(=O)C(C)OC)c2ccccc12 C(=O)(C(C)(C)C(O)C(C)C)N.C(C(C)(C)CN(C)C(C1CSC1)=O)OC C(c1cccc(Cl)c1)=C(C)C(=O)NC1(CCNC(=O)CCC(C)(F)F)CCCC1 C(=O)(CC1=NNC(=O)C1)N(C1CCCC(NC(=O)CCCc2n[nH]c(=N)s2)C1)C Cc1ccc2cc(C(N3CCCC3C(N3CCC(O)CC3)=O)=O)sc2c1 N1(C(CCCN(C)C)=O)CCC(C)(C)C1C(=O)NCCC(O)CO Cc1ccc(NC(=O)CN2C(=O)C(=O)N(C)C2=O)c(F)c1 O(S(=O)(=O)c1ccc(NC(C)=O)cn1)c1c(OC)nsc1 c1(C(=O)NCC2(F)CCN(C(C(c3n(C)ccc3)=O)=O)C2)cccc([N+](=O)[O-])c1 C(CC(=O)NCCCCN1CCCC1)N(C(C1CC1Cl)=O)CCO CC1CN(C(=O)CSCc2ccc(F)cc2)CCN1C(c1ccc(O)nn1)=O C(=O)(C1CNc2ccccc21)NCC(C)N(C(CC(CC)C)=O)C c1(C(C(=O)NC(CNC(CCNC(COC)=O)=O)C2CC2)O)cc(Cl)ccc1F C(=O)(CC1COCc2ccccc21)NCC(C)(C)NC(CC1CCN(C)C1)=O C=CCC(C(=O)N1CC(NC(C2CCCCCC2)=O)C(SC)C1)C(C)(C)C CC1CC(C(=O)NCC2CC(NC(=O)CC(F)(F)Cl)C2)CC(C)(C)C1 CC(C)CC(O)C(=O)NCc1ncoc1C1CN(C(=O)CC(C)CF)C1 c1(C(=O)OC)cc(S(=O)(=O)NCC2CC3(C2)CC32CC2)cc([N+](=O)[O-])c1C c1(C(=O)NC2C(OC)CN(C(C3(CC)CC3)=O)C2)cc(OC)ccc1OC C1(N(C)C(C2CSC2)=O)CCN(C(c2cn(CC(N)=O)nn2)=O)C1 C(C(C)C(F)C(=O)NCCCc1ccnn1C)NC(Cn1c(C)nnn1)=O C1(C2(C(=O)NCC(CNC(=O)CCn3cccn3)F)CC2)CCCCO1 C12(C(N3CC(O)(CCNC(=O)CC4CCCC4O)C3)=O)CC(CF)(CO1)C2 Cn1cc2cccc(C(N3CC4CN(S(=O)(=O)c5nccs5)CC34)=O)c2n1 Cc1cncc(C(=O)NC(C)Cn2cc(CCOCC3CCCOC3)nn2)c1C c1(C(=O)NCCCCN(C)C(C2CC2(F)Cl)=O)nn(C)cc1Br Cc1ccn(CC(N2CCCC(N(C(=O)CSCCN(C)C)C)C2)=O)c(=O)c1 c1(OC)ncccc1S(=O)(=O)N1CCC(NC(c2cnc(N(C)C)o2)=O)C(F)C1 c1(C(=O)NCC2CCC(C(N)=O)CC2)c(Br)nc2n1CCCC2 C1(NC(C(C(C)C)NC=O)=O)CN(C(c2cc(Br)n(C)c2)=O)CC1N=[N+]=[N-] c1(CC(N2C3(CNC(C(C)=CC)=O)CC(C2)C3)=O)cccc(Cl)c1OC N1(C(CCn2ncc(C)c2)=O)CCC2(CCCCC2NC(C2CCC2)=O)C1 C(C(C)CC(=O)NCCC1(C)CC1)NC(C=CC(C)(C)SC)=O CC1CN(C(=O)C(=O)NC2CCN(S(C)(=O)=O)CC2)CCN1C(=O)C(C)C(F)F N1(C(C(CSC)(C)NC(=O)C(F)CC(C)(C)C)=O)CCC2CN(C)CCC12 c1(C(=O)NCCCC(C)(C)NC(C(C2CC2)OC)=O)ccc2nnn(O)c2c1 c1(CCC(=O)OC)nc(-c2cccs2)no1.N(CC)(CC)CC c1(C(C)(C)C)ncc(C(=O)NCC(C2CCC2)NC(c2n[nH]cc2Cl)=O)cn1 c1(NCC(N2CCC(C(CNC(CCC#C)=O)O)CC2)=O)c(F)cc(C)cc1Cl C1(C(N(C2CCCC(O)C2)C)=O)CC(C)(C)CN1C(=O)CC1OCCC1(C)C N1(c2c(C(F)(F)F)cc(Cl)cc2)CC2C3CCC(C3)C12 C1(NC2CCCCCC2)CCCCN(C(=O)NC(C(F)(F)C2(OC)CCC2)=O)C1 c1(C(N2CC(C(C)C)C2)=O)cncc(CNC(=O)C(c2cncnc2)C)c1 C1(NC(COC)=O)CN(C(C2CC(SC)C2)=O)CC1C(F)F.c12cccc(n1)O2 C12(NC(c3cc(CC4CC4)c[nH]3)=O)CCCC1CN(C(C1CC3CCC3C1)=O)C2 C(=O)(C(C)CCCOC)N(CCCNC(C1(C=C)CC1)=O)C1CC1 N12CCCC(CC1)CC1CC1C2=O.N1(CC)CCCC(NC2(C#N)CCCC2)C1 C1(C(=O)NCC(CC(C)C)(C)NC(=O)CC(C)(F)F)CCc2c(ncn2C)C1 C1(NC(C2N(C(C3(C)COC3)=O)CC2)=O)CONC1=O C1(C(=O)OC)CC2CC1CC2N(c1sccc1NC(=O)OC)C.C1(C)CN1C c1(CC(=O)N(CC(C)N(C)C(c2cccc(CC#N)c2)=O)C)ccc(F)c(Cl)c1 CC(N=c1nc(N(C)CC2CC2(F)F)c2c([nH]1)COC2)c1ccoc1 N1(C(CCOCCOCC)=O)CCC(C)(NC(c2ccn(CCF)n2)=O)CC1 C1(NC(C(C)(C)c2cscn2)=O)CC1C1CCN(C(C2(C)CC=CCC2)=O)CC1 Cc1cc(F)c(F)cc1NC(=O)CN1CCN(C(c2cnc(Br)s2)=O)CC1 C1CCN(N2Cc3ccoc3C2)CCO1 c1(N(CCCNC(C(C)CC(N)=O)=O)C)nc(Cl)nc2cnn(C)c12 CN1CCN(C(c2sccc2N(C)C)=O)CC1c1ncc[nH]1 N1(C(CCOCC)=O)CCC2(CC2C(=O)NCc2nccs2)C1 C12(C(N3C(C(=O)NC4CN(CC(F)(F)F)C4)CC3)=O)C(NC(N)=O)C3CC1C2C3 C1(C)(NC(C2C(=C)C2)=O)CCN(C(c2oc(C(F)F)cc2C)=O)CC1 N1(C(COC)=O)Cc2cnn(C3CCN(C(C4C(C(F)F)C4(C)C)=O)CC3)c2C1 c1(NC(C2CC3(CN(C(C(C)(CO)CO)=O)C3)C2)=O)c(F)cc(I)cc1[N+](=O)[O-] Cc1cnc2n1CCC(CC(=O)NC1(Cc3ccccc3)CN(CC(F)F)C1)C2 CCCC(C(=O)N1CCCC1CCCNC(=O)CC1CC2CC2C1)OC c1(NC(C23C(CN(C(CCC)=O)C2)C3)=O)ccc(OC)c(C)c1 CC1=NOC(C(=O)NC2CCN(C(c3[nH]nnc3C)=O)C2)C1 C1(NC(C(C)NC=O)=O)CCC2CN(c3cc(-n4ccnc4)ncn3)CCC2C1 C(CC(=O)N1CCC(C(=O)NCc2ccc(F)nc2F)O1)OCCC NS(=O)(=O)c1ccc(CC(=O)NC2CCC(CNC(C3COC(=O)N3)=O)C2)s1 Cn1ncc(CNC(C2CC2F)=O)c1C(=O)NCCOCC(F)F Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2ccc(Cl)cc2Cl)nnc1C C12(CC#C)CCN(C1)C(=O)OCCNC2=O.c1(CC)cn(C2CC2)cn1 c1(CN(C(C2CCCC23CC3)C(=O)NC(CC)(C)C)C)ccc(OC)c(Cl)c1 c1(C(=O)NCC2CCC(NC(CC(=O)NCC)=O)C2)cc(C)c(O)c([N+](=O)[O-])c1 c1(C(N(C(C)CCNC(=O)CSc2nc[nH]n2)C)=O)c(O)cc(Cl)cc1F Cn1c(C(=O)NCCC2CCCN2C(C2CC(O)C2)=O)cc2sccc12 c1(N2CC(CCC)C(N(C)C)C2)[nH]c(=NCN(C)C(C)=O)nc2sccc12 CCC(C)C(C(=O)NC12CCC(C(=O)NCC(C)NC)(CC1)C2)N(C)C c1(C(=O)NCC(=C)CCNC(=O)CCC=C(C)C)cc2ncccc2cc1Cl C12CCN(CC1)C(=O)C(C)OC2.c1(C(=O)OC)nc(CN)oc1C C#CC12CC(CN1C(=O)C1=NOC(CNC(C3CC(C)=NO3)=O)C1)C2 C1(CC(=O)NCCN(CCC)CCC)CCCC1C(=O)NCC C(=O)(C(C)(C)CCSC)N1CCN(CC)CC1.n12cc(nn1)C(SC)OC(=O)C2C C1(NC(CC(CC)C)=O)CN(C(=O)NC2(Oc3cccc(C)c3)CC2)CC1(C)C c1(C(=O)NC2C(C)CN(C(C3CCN(C4CC4)CC3)=O)C2)c[nH]c2c(Cl)cccc12 c1(C(=O)Nc2cn(CCCOc3c(C)n[nH]c3)nn2)ccc(C(=O)O)c(O)c1 CC1CCCC=C1C(=O)N(C)CC1(O)CN(C(=O)COc2ccccc2)C1 N1(C(c2c(C)cccc2)=O)CC(C2CCCCN(C(C3CCCS3)=O)C2)C1 N1(C(=O)NC(c2cscn2)C)CCn2cnc(C(N)=O)c2C1 CN1C2CCC1CN(c1cc(NCCC3(C(F)(F)F)CC3)nc(C(F)(F)F)n1)CC2 C(=O)(C(CNC(=O)CCc1ccncn1)CC1CC1)NC(C)Cc1cncnc1 S(=O)(=O)(c1cnccc1N1CCCC(C#N)C1)NCc1ccc(CC)o1 Cc1ccc(NC(=O)C(C2CC2)N(C)C(c2cccc(Cl)c2)=O)c(CO)c1 C1(N(C(c2ccc(C(N)=O)s2)=O)CCF)CCCN(C(=O)Cc2sccc2Cl)C1 c1(CNc2cccc(C(=O)NC(C)C)c2)ccc(O)c2ccccc12 C(CCC)(C(=O)NC(CCF)C(=O)NCC1(CC2CCC2)CC1)=CCC C1(C)(C(=O)NCC2CCC(NC(CCC3CC(OC)C3)=O)C2)CNC(=O)C1 Cc1cc(C(N2CCC(OCc3ccc(C)o3)C2)=O)n(Cc2ccccc2)n1 c1(OC)ccnc(C(=O)NCCCNC(c2coc(C(F)F)c2)=O)c1N c1(C(N2C(CNC(C3CC(SC)C3)=O)COCC2)=O)ncc(C)cc1C N1(C(C(C2CCCC2)OC)=O)CCN(C(=O)C(C)OC(C)=O)CC1 C(=O)(C1=CCCC1(C)C)N1CCC(NC(c2cncc(OC)c2)=O)C12CC2 CC(C)(C#N)CCC(=O)N1CCC(CCNC(C2(C)CC2c2ccccc2)=O)C1 c12ccc(nn1)N1CC(CC1)N2.c1(C(N2CCOCC2)=O)ncncc1Cl N1(C(c2c(CC=C)cccc2)=O)CCOC(C(=O)NCCC2=CCCCC2)CC1 CC1(C)CCN(C(=O)C(O)c2cnc[nH]2)CC1NC(=O)CCOCC(F)F CCC(C)(CNC(=O)CCC1(NC(C2CCC(F)CC2)=O)CCCC1)C(N)=O C1(C)(CNC(C(CO)OC)=O)CCCN(C(c2cc(C)sc2C)=O)C1 N1(C2(C(=O)NCCN(C(=O)CSC3CCCC3)CC)CC2)CCOCC1 c1(CNC2CCN(S(CC)(=O)=O)C2)ccc2c(C)[nH]nc2c1 C1(C)(C(N(C2CC2)CC2C(C)OCC2)=O)CCN(C(=O)CC2CCCC3CC23)C1 c1(C(N(CC(C)NC(c2cncc(C)n2)=O)C)=O)sccc1S(=O)(=O)NC1CC1 c1(CC(N2CCC(NC(C(=O)NC(C)C)=O)C2)=O)ccc(C(F)(F)F)nc1 C1(C2C(NC(CC3CN(C(C)=O)C3)=O)C2)CCCCN1C(c1cnn(C)c1)=O n1(CCCOC)nc(COCC(=O)NCC(CO)NC(=O)C2=COCC2)ccc1=O C1(C(=O)NCC(CN(C)C(c2csc(C(F)F)n2)=O)O)Cc2cc(Cl)ccc2O1 N1(C(c2ccc(CN(C)C)cc2)=O)CCN(C(=O)Cc2ccn(C)n2)C(CO)C1 C#Cc1cccc(C(N2CCCC(C(=O)NCC(C)C(F)F)CC2)=O)c1 c1(OC)cc(C(=O)NC(CNC(c2nc(C)oc2C)=O)CO)ccc1[N+](=O)[O-] C1(NC(C(CC)C)=O)CC(C(=O)N2CCCC3(C2)N=N3)=CC1O C1(CCNC(C2CCCCS2)=O)CCCN(C(=O)C=CC2CCC2)C1 N1(C(Cc2ccc(C)s2)=O)CC(CNC(C2CCCS2)=O)CC(C)C1 C(=O)(CCCCCNC(C1(C)CCCC1C)=O)NC(CCC(=C)C)C c1(NC(C)=O)nc(C2CCCC(NC(=O)C(=O)N(C)C)CC2)cc(O)n1 c1(C(=O)NC2C(C)N(c3nnc(C4CC4)s3)CCC2)c2c(c[nH]c1=N)CCC2 c1(C(=O)NCC(C2CCC2)NC(=O)CNC(N2CCCC2)=O)cnnc(O)c1 C1(C2C(CC(=O)N(C3CC(C(=O)OC)C3)C)C2)CCCCO1.C1CO1 c1(N2CCN(Cc3ccc(C#N)nc3)C3C2C3)ncc2ccc(F)cc2n1 N1(C(CSCCN(CC)CC)=O)CCC2CN(C(C3CCCC3)=O)CC12.C(C)OC N1(CCn2c(N)c(C(=O)O)cn2)CCC2C(=O)NC(=O)C2C1 C(=O)(C1=CCCOC1)N1CC(F)(CNC(=O)CCCn2cncn2)C1 c1(C(=O)NCC2C(C)CCN(C(COCCCOC)=O)C2)sc2cncn2c1C C12(C(N3CCC(NC(c4cc(F)cs4)=O)C(F)C3)=O)CCCCCC1OCC2 C1(CC(N2CCC(CN(C(CC3(OC)CCC3)=O)C)C2)=O)C=NN(C)C1=O c1(C(=O)NC2CN(C(CC(C)OC)=O)CC2C)cc(N(C)C)cc(Br)c1 N(C(=NCCCC1CC1(C)C)NC1CN(C2CC2)CC1C)Cc1c(C)ncs1 c1(CC(=O)NCCC(C)NC(C2CCCC2(F)F)=O)ccc2c(c1)CCCN2C N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CC2(CCN(C(=O)C=CC3CCOC3)C2)C1 Cc1nc(C)c(F)c(=NCC(C)CNC(=O)C(O)C2CCCC2)[nH]1 C(=O)(CCCCCC1CC1)NCC(C)NC(c1cn(CC2CCCO2)nn1)=O N1(C(=O)Nc2noc(CC)c2C)C2CCC1CN(C(=O)OC(C)(C)C)CC2 Cc1cc(N(C)CC2CCOCC2)nc(=NCC(C)c2ccc(Cl)cc2)[nH]1 c1(C(N2CCCC(C(C)C(=O)N(C(C)CN(C)C)C)C2)=O)cncc2[nH]ccc12 C1(C)(C(N2CCC(C(C)NC(c3c(C)c[nH]c3)=O)CC2)=O)CCCCNC1=O N1(C(c2cc(CCNC(c3nc(C)oc3)=O)on2)=O)CC2(CNC(=O)C2)C1 C1(NC(c2c(CC)nn[nH]2)=O)CCN(C(=O)CSc2n[nH]c(=N)s2)CC1F C1(NC(Cc2c(C(C)C)con2)=O)CC12CCN(C(c1cc(Cl)cs1)=O)CC2 c1(C(N(CCCNC(c2c(COC)scc2)=O)C)=O)n[nH]c2ccc(CO)cc12 c1(C(=O)NC(C(C)C)CNC(=O)CC2CC2(C)C)cc(F)cc(Br)c1O C(CC(C)C(=O)NCC(O)CNC(c1onc(C)c1C)=O)=CCC N1(C(C2(C)CCC2)=O)CCCC(C2CCN(C(=O)CC3CCCOCC3)C2)C1 CN(C1CS(=O)(=O)c2ccc(Cl)cc21)CC(=O)C(F)(F)CCl N1(C(c2ccc(CC)s2)=O)CCC2CN(C(c3ccc(Br)o3)=O)CCC2C1 Cc1ccc2c(c1)C(C(=O)NCC1(NC(=O)CC3C=CCC3)CC1)CC2 C=CC(C)(C)C(=O)NC1CC(NC(c2cnn(C(C)CC)c2C2CC2)=O)C1 C1(NC(CS(C)(=O)=O)=O)CC2(CCC(NC(C(=O)O)C(=O)O)OC2)C1 Cn1cc(C(=O)NCCCNC(=O)CN2CCC(C(N)=O)CC2)c(O)n1 CCCS(=O)(=O)CC(=O)N1CCC(NC(=O)CC2CC3(CC3)C2)C(CO)CC1 N1(C(=O)OC(C)(C)C)CCC2(CC1)CC(NC(Cc1cccs1)C(=O)O)CO2 c1(CC(=O)NC2CC(CNC(c3c(C)ccc(O)c3)=O)C2)ccc2c(c1)COC2 c1(C(=O)NCc2ccc(CNC(C3(C)C(C)(C)C3)=O)cc2)cccc2cncn12 C12(NC(CCc3ccc(C)o3)=O)CCCC1CN(C(c1cc(C(F)F)no1)=O)C2 c1(C(CC)C(=O)NC(C)(CNC(=O)CSS(C)(=O)=O)C2CC2)ccc(Cl)cc1 C1(OC)CCn2cc(C(N3CCCC(CNC(C4CS(=O)(=O)C4)=O)C3)=O)nc2C1 C12(NC(C(N3C(CC)CCC3)=O)=O)CCC1CN(C(=O)Cc1ccc(F)cn1)C2 N1(C(C(C(CC)O)C)=O)CCC2(CC1)CN(C(=O)CS(=O)(=O)CCO)CC2CO c1(C(=O)NCC2N(C(C(C=CC)O)=O)CCCC2)ncc(F)cc1F C1(NC(C=CCCC(C)C)=O)(CO)CCCN(C(=O)C(C)C2CC2)C1 c1(CC(C(=O)N(CC(C)NC(COCCC=C)=O)C)O)c(F)cccc1Cl O=C(C#CC1CCOC1)NC1(CNC(=O)C2=CCSC2)CCOCC1 C1(C(N(C(C)CCNC(=O)CSC(=N)N)C)=O)Cc2ccccc2CO1 C1(C(=O)NC2(CNC(c3cc(OC)c(O)nc3)=O)CCC2)CCCC2(CCC2)O1 Cc1cc(=O)n(CCC(=O)NCC2CCC(F)(CNC(=O)C(C)(C)CO)C2)cn1 c1(CCNC(c2ccncc2Cl)=O)ccc(CNC(C23CCC(C2)C3)=O)cc1 c1(C2(C(=O)NCCC3(O)CN(C(=O)C=C4CCC4)C3)CC2)ccc(F)cc1F CCC(C)(CNCC1CCC(O)CC1)C(=O)N=Cc1cn(C)nn1 c1(C(N(CCN(C(C2C(C)C2)=O)C)C(C)C)=O)cccc(-c2cccc(Cl)c2)c1 c1(CC)cc(F)cc(Br)c1.Cc1nn(C2CC2)cc1C(N)=O c1(C(N2C(CNC(C3CC(F)(CO)C3)=O)CC(OC)C2)=O)cc2cccnc2s1 c1(C(=O)NCCCN(CC)CC)cc2nc(C)cc(C(F)(F)Cl)n2n1 c1(C(=O)NCC2(C)CCN(C(C)=O)C2)ccccc1S(=O)C(F)(F)F C1CCC12CCNCC2.c1(-c2nc(N3C(=O)OCC3)on2)cccn2ccnc12 c1(OC)ccc(C)c(C(=O)NCC(C)(C)CNC(=O)Cn2cc(C)ccc2=O)n1 c1(C(=O)NC2C(CC)CN(C(C3(CC(C)C)CC3)=O)CC2)c(N)cc(F)cc1F C=CCCCC(C(=O)NCCC(F)(F)Cl)NC(C1CCCCC1(C)C)=O CC1C(NC(=O)C(C)N(C)C)CCCN1C(c1ncoc1C(C)(C)C)=O N1(C(C2C(C)CC(C)O2)=O)CCC2(C1)CN(c1nc(C3CCCC3)ns1)C2 S(=O)(=O)(c1ccc(NCC(CC)n2cccn2)c(F)c1)N1CC(CC)OCC1 c1(C(C(=O)NCC2(O)CN(C(c3c(C(C)C)con3)=O)C2)(C)C)cccc(F)c1 C(=O)(CCCC(C)(C)NC(=O)CN(C)C1CC1)NC(CC#CC)C C(=O)(CC(C)C(=O)NCc1cc(C(N2CCNC(=O)C2)=O)ccn1)OC c1(CNC(c2oc(C(=O)OC)c(C)c2)=O)cnn2c1CN(C(C1(F)CC1)=O)CC2 c1(C(=O)NC(C(=O)NC2(CSC)CCC2)C2CCCO2)ccc(O)cc1F C1(N2CCC(OC)CC2)CCC(N=c2nc(NCC(C)O)c3nc[nH]c3[nH]2)CC1 c12ccc(c(C)c1)[nH]c2=O.C(=O)(CCCCC1CC1)NCC1C(COC)CCC1 Cc1ccn(C(C)C(=O)N(C2CC(C(=O)N(C)CC3(CC(C)C)CC3)C2)C)n1 c1(CC(=O)NCC(COC)C)cc(Cl)ccc1C C(=O)(C1=C(C)OCCC1)N(CC(C(=O)NCC(C)NC(=O)OC)(C)C)C C1(NC(CCC=C)=O)(CO)CCCN(C(=O)COCC(=O)OCC)C1 C(N=c1[nH]cnc2[nH]ccc12)C1CC(COC)CN1c1cc(F)ncn1 C1(NC(c2scc(OC)c2)=O)CCCC12CCN(C(c1cc[nH]c1C(C)C)=O)C2 C1(C(=O)NCC2C(NC(C3(SC)CC=CC3)=O)CCC2)CCCN(C(C)C)C1 N1(C(c2cc(C)[nH]c2)=O)CCC(F)(F)C(CNC(c2nccc(CO)n2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1CC(CC(CNC(C(C)SC23CC(C2)C3)=O)(C)C)C1 N1(C(c2cn(C(C)C)nn2)=O)CC2CC(NC(=O)CSCc3cscn3)CC2C1 C(=O)(C1CCc2ccccc21)N1C(CN(C(c2ns[nH]c2=O)=O)CC)CCC1 C1(O)(CNC(c2cnc(CC(C)C)s2)=O)CCN(C(=O)C(F)=CC2CC2)C1 c1(C(N(CCC(C(C)C)NC(=O)C#CC(=O)N(C)C)C)=O)cccn2ncnc12 N1(C(C(C)(CO)NC(C(CCCC#C)C)=O)=O)CC2(CCC(O)CC2)C1 N1(C(CC=C)=O)CC2CC1CN(C(=O)C=CC1CCOCC1)C2 C1(C(=O)NC2(CC)COC2)CCC(n2cc(CC(=O)O)nn2)C1 CC(C)(C(=O)N1CCN(CCc2cn(-c3c(F)cncc3Cl)nn2)CC1)C(F)F C(=O)(C(O)P(C)(C)=O)NC1(CCOC)CCN(C(=O)CCN2CCCCCC2)C1 c1(N2CC3C(C)C3C2)[nH]c(=NCCC2CCCCO2)nc2scnc12 C1(CNC(C(CC2CC2)OC)=O)CCCCCN1C(c1cc(=O)n(C)cn1)=O c1(C(=O)NC(C(CO)NC(CCCc2c(C)ccs2)=O)C)ccc(CSC)cc1 O=C(C1=CCS(=O)(=O)C1)NC1CC(CNC(c2cnn(C3CCC3)n2)=O)CC1O C1(C(=O)NCc2cnc(C)o2)CCN(C(=O)C2CCC3(CCC3)C2)O1 C1(CNC(C(=Cc2ccccn2)C)=O)C2CCC(C2)N1C(C1CN2CCC1C2)=O C1(C#CC(=O)N2CCCC(C(=O)NCCC[Si](C)(C)C)C2CC)(CC)COC1 N1(CCC(=O)NCC2CN(C(=O)CC3CC3(Cl)Cl)C2)CCCCC1=O CC#CCC(C(=O)NCC(C)C(C)CC)NC(c1n[nH]c(C)c1Cl)=O N1(C(c2cnc(COC)s2)=O)CCCC2(NC(=O)Cc3cc(C)no3)CCCC12 c1(O)ccc(Br)cc1CO.N1(CCCN(C(=O)NC2(OC)CC2)C)CCN(C)CC1 CC(C)C(F)(CNC(c1cccc(F)c1F)=O)C(=O)N1CCC(O)(C(N)=O)C1 C1(C(=O)Nc2ccc(CC)cn2)CCN(C(=O)C(O)C2CCCC2)CC1O C#CC1CN(C(C2CCC(=O)N2)=O)CCN1C(=O)CCC1CC1(F)F c1(C(=O)NC2C(C=C)CN(C(C3CNC(=O)N3)=O)C2)nnc2ccccc2c1N C12CN(CCCO1)C2.Cn1ncc(Cl)c1CC(=O)Nc1ncc(C(C)(C)O)cn1 c1(C(=O)NCC2(F)CCN(C(C=CCOC)=O)C2)cccc([N+](=O)[O-])c1Br C1(C(NOCCCN(C)C)=O)CCCCC1NC(C1CC(=O)CCO1)=O C=CCCCC1C(=O)N2CC(O)(C2)C(=O)NCC(=O)N1.C(CC)SC c1(OC(C)C)ccc(C(N2CCC(O)(C(C)CNC(=O)CCCF)C2)=O)cc1 C1(CC)C(C(=O)NC(COC)C2CC2)CCN1C(c1nnsc1C)=O Cc1ccc2n[nH]cc2c1C(=O)NCC(O)CNC(=O)C(F)(F)C(C)O c1(C(N2CC3C(COC(C)(C)C)C3C2)=O)c[nH]c2ccncc2c1=O C1(C(=O)OC(C)(C)C)OCCC1NC(C1(CSCC(F)(F)F)CC1)=O C=CCCC(C)C(C(=O)NC1CC1)N1CC(C)OC2(CCOC2)C1 C(CN(C1CCOCC1)N(CC(F)(F)C1CC1)C1CCCC1)OC(C)(C)C CC(=O)CCCC(=O)N1CCN(C(c2cccc(CN(C)C)c2)=O)C2CC12 C1(OC)CN(C(=O)Cn2ccc(C(N)=O)n2)CC1NC(=O)C(C)SC(F)(F)F c1(C(=O)NCC2(CNC(C(CC#C)O)=O)CCCC2)ccn2c(O)nnc2c1 N1(C(C(CCC=C)NC(=O)CC(C)C=C)=O)CCC2CCC(C1)N2C c1(OC)ccc(C(=O)N(C2CCCC2)CCNC(=O)C2=CCCC2C)cc1F c1(CC)cccc(C(N2CC(CO)(NC(=O)C=Cc3ccc(Cl)cc3)C2)=O)c1N c1(CC(=O)N(C(C)CNC(=O)CC2(O)CCCCC2)C)c[nH]c(=N)nc1O C1(CC(=O)NCc2c(C(N(C3CCCCC3)C)=O)cco2)CCC(=O)NC1 C1(c2cc[nH]n2)(C(=O)NC2(C)CN(C(C=CC(C)=O)=O)C2)CCOCC1 Cc1ccc(Cn2nnc(N3CCC(C)(NC(=O)C#CC4CC4)C3)n2)cc1 N1(C(c2n(CC#C)ccc2)=O)CCCCC1C1(N(C(C2(C)CC(=C)C2)=O)CC)CC1 c1(C(=O)NC2CC(NC(C3C(OC(C)=O)C3(C)C)=O)C2)c(C(F)(F)F)noc1C C1(OCC(=O)NC2(CC(F)CO)CC2)CCN(C(c2csc(O)n2)=O)C1 c1(C(N2CC(C#CC)C2)=O)cc(OCC)cc2ccoc12 c1(OC)cc(CC(=O)NC2CCCN(C(c3nccnc3N)=O)C2C)cc(F)c1 C1(NC(COCCSC)=O)CC2(CCN(C(=O)C(C(C)C)c3ccncc3)C2)C1 C12(CCCCC1)CC(=O)NC2.c1(CCN(C(=O)CSC(F)F)C)cn(CCO)nn1 N1(C(CONC(=O)OC(C)(C)C)=O)CCCC12CCN(C(=O)CP(C)(C)=O)CC2 c1(C(C(N2CC3(C(C(=O)Nc4c(C)nn(C)c4)C3)C2)=O)C)ccc(O)c(O)c1 C#CCCCCC(=O)N1CC=CC(C(=O)NCCC)C1 C1(=O)CC(=O)NCCCN1C(C)C.c1(CSCC(=O)NC(C)=O)cccs1.CO n1(CC(=O)N(CC(C)O)CCNC(=O)CCCc2ccsc2)cccnc1=O c1(C(N2CCC3(NC(C=CSC)=O)C(C2)C3)=O)sc2ccccc2c1Cl c1(CC)ncc(C(=O)NCCC(C)N(C)C(c2cnnn2C)=O)s1 C12(C(N3CC(C)OCC3)=O)CC(CO1)N(C(=O)CC(=O)N(C)C)C2 C(=O)(C(CC)C(=O)N1CC(CC(F)C(N2CCCC(N(C)C)CC2)=O)C1)OCC C1(NCC(N2CC(NC(=O)CSCC(F)F)C2)=O)CCC(O)CC1 c1(C(N(CC(C)(C)CNC(=O)C=CC2CCCC2)CC)=O)cccc(CCO)c1 C1(CC(=O)OC)CN(C(=O)NC23CC(C2)C3)CC1C c1(CN(C)Cc2ccc(F)cc2CO)ccc2c(ccn2C)c1 N1(C(CNC(CCC2CC(=C)C2)=O)C)CCN(C(=O)C(C)SC)CC1 C#CCC(CC#C)C(=O)N1CC2(CC2)CC1CNC(C1(C2CC2)CC1)=O N1(C(Cc2cc(C)sc2)=O)CC(C)(C)OCC1CNC(=O)COC1CCCC1 c1(CC)ccc(CN=c2nc(-c3ccccc3)o[nH]2)cc1C Cc1cc(F)cc(C(N2CCOC(CCNC(=O)CCCCN(C)C)C2)=O)c1C CC1(CC(N2CCOCC(NC(C3CCCCC(=O)N3)=O)C2)=O)CCCCCC1 C1(CNC(C2(CC=C)CC2)=O)C2CN(C(=O)CSCC)CC12 C1(C(=O)NCC(CC)O)CN(C(=O)C(O)CN(C)C)CCO1 C=CCC(C)C(=O)NCCN(CCOCCO)C(c1coc(C2CCC2)n1)=O CC1=C(CNC(c2ncsc2C)c2nnnn2CC2CCCO2)CCC1 N1(C(CSCC(C)=O)=O)CCC(C2(NC(=O)CCc3cncc(F)c3)CC2)C1 C(=O)(C(CCCCC1CC1)N(C)Cc1ccc(Cl)s1)NCCOC C(C(C)(C(=O)O)NC(c1ncn(Cc2ccccc2)n1)=O)NC Cc1nn(C)c(C)c1CCC(N1CCCC1C(C)(C)NC(CC)=O)=O.c1(C)ccsn1 c1(C(=O)NC2CC(NC(C3(N(C)C)CCCCC3)=O)C2)cc2ncn(C)c2cn1 Cc1ccc2c(=NCC3CC4(CC4)C3)c(N3CCOCC3)c[nH]c2c1 N1(C)Cc2c(F)ccc(F)c2C1.C1(NC(=O)O)CC(CNC(C(C)(C)C)=O)C12CCC2 CCCC(C#N)C(=O)NC(CC1CC1)C(=O)NCc1ccnc(F)c1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)c2cccs2)=O)nccc2ccncc12 C1(C(=O)NC(C)CCNC(C2(c3ccccc3F)CC2)=O)CCOC2(CCC2)C1 c1(C(=O)NC2C(OC)CN(C(=O)CC3CCC3C)C2)c(N)c(F)cc(F)c1F c1(NC(C)(C)CNC(C2CCC(C(N)=O)C2)=O)ccc2c(n1)CCC2=O c1(C(=O)OC)ccc(C=CC(=O)NCC2CC(F)(CNC(=O)CSC(F)F)C2)o1 c1(C(N(CCN(C(C(CCC)O)=O)C(C)C)C)=O)cc(C)cc2cnnnc12 c1(NC(C2C(NC(c3cc(CC)no3)=O)C2)=O)ccc(Br)cc1C(N)=O C1(C(=O)NC2C(CNC(COc3cn(C)nc3)=O)CC2)CC2C=CCC(C1)C2 c1(CNC(C(=O)NCC(C)(C)C2CCCO2)=O)ccc(-n2cc(Cl)cn2)cc1.NCC C=CCC(CC)C(=O)NCC(C)C(=O)N1CC(C)(CF)C1 C1(CNC(=O)C=CCc2cccs2)CN(C(=O)COCC2CCOC2)CC12CC2 N1(C(C2C(CNC(C3N(CC)CCCC3)=O)CC2)=O)CCC2(CNC(=O)C2)C1 C=CCCCCCCCC(=O)N(CC(C)CNC(c1cccn2nnnc12)=O)C N1(C(CN(C(c2c(C)scc2)=O)CC2CC2)=O)CC2COCC2C1 C(=O)(C(C(C)NC(C1CCNC1=O)=O)C(C)C)N1CCC(O)(CCC)CC1 C(=O)(C(C(C)C(C)(C)C)N(C)Cc1ccc(Br)s1)NCc1c(OC)cccc1 C#CCCC(O)C(=O)N1CCC(CO)(NC(c2cc[nH]c2)=O)CC1 Cc1cccc(C(C)NC(C2(CNC(=O)CCn3cccn3)CC(C)(C)C2)=O)c1 C(C(C(=O)N1C(COC)CC1C)C(C)C)NC(C1C(CCOC)C1)=O Cc1c(C(=O)NCCC(C)NC(c2c[nH]nc2C(F)(F)F)=O)oc2ccccc12 C=CC(F)(F)C(=O)NC(C)CCC(=O)NC(C)CCCCCOSC c1(C(=O)NC2C(CNC(C(CSC)(C)C)=O)C2)ccc(C)c(C#N)c1 c1(C(=O)NCC(C)NC(CCCCOC)=O)nc(Br)n2c1CCCC2 C(=O)(C(C)(C)CC(=O)NC(C)CCN(C(=O)CC(C)NC(N)=O)C)OCC C=C=CCCC(=O)N(C)CCNC(=O)CC1CC(=O)NC1=O C1(CNC(C2N(C(CC3(OCC)CC3)=O)CCCC2)=O)CCCC12CCC2 C1(C(N2CCC(C(N3CC(C(=O)OC)C3)=O)C2)=O)CCCN(C(C)=O)C1 C(=O)(CCC(Cl)Cl)NC(CC(=O)OCC)c1ccccn1 C1(NC(c2nc(C(C)C)oc2)=O)CCC(N(C(=O)CC2CN(C)CCO2)C)CC1 C(=O)(CC(O)CC(C)(C)C)N1CC(CC(=O)OC)OCC1.C12(O)CN(C1)C(=O)C2 CCCCCCC(=O)NCC1CC(F)(CNC(=O)CC=Cc2ccccc2)C1 Cc1cc(F)c(C(=O)NCC2CCC(NC(=O)Cn3ncnn3)C2)cc1Br c1(NCCC(=O)NCC)[nH]c(=NCC(C)(C)c2n[nH]c(CC)n2)nc2sccc12 C1(c2n(CCOC)nnn2)(NC2CC(CC3CC3)C2(C)C)CCS(=O)(=O)CC1 c1(CC(=O)NCCCN(C(c2c(C(=O)OC)coc2)=O)C)nnc(C)n1C C1(C(=O)NC(C=C)C2CC2)C(O)CCN1C(=O)C(c1ccoc1)OCC C(=O)(C(C)CC(F)(F)F)N1CCC(O)(CNC(Cc2cn(C(C)C)nc2)=O)C1 C=C1CC(C(=O)NC(c2ccccc2)C#N)N(C(C2CCNC2=O)=O)C1 C1(C(=O)NCc2cn(CC=C)nn2)CC12CCN(C(c1ccc(CO)cc1)=O)C2 N1(C(C2C(C)C2C)=O)CCC(C2(NC(=O)Cc3nncs3)CC2)CC1 n1(CC)ncc2c(NC3CC(NC(C4CCC5CC5C4)=O)C3)ncnc12 n1(CCOC)cc(NC(c2conc2CNC(C2CCC(O)C2)=O)=O)cn1 C1(CNC(C(C)SCC)=O)CCC2CN(C(=O)CC3CC(C)=NO3)CC12 C1(N(C(c2ccn(CCC)n2)=O)C)CN(C(c2cn(CCO)nn2)=O)CC1F C1(NC(CCc2onc(CC)n2)=O)CN(C(=O)C=CCO)CC2(CCOCC2)C1 C1(NC(c2cnc(SC)s2)=O)CCN(C(c2cccc(SC(C)C)c2)=O)CC1C N1(C(c2nc(CC)[nH]n2)=O)CCCC(C(N2CCC(C(N)=O)CC2)=O)C1 c1(CC)occ(C)c1C(=O)NCCc1nocc1C(=O)NC1(CC2CC2)CCC1 C1(N(C(C(c2scc(CC)n2)(F)F)=O)C)Cc2cccc(OC)c2C1 N1(C(CC2CC3(CN(C(c4ccon4)=O)C3)C2)=O)CC2CCCCCCC12 Cc1cc(C(N2CCC(NC(c3cc4c([nH]3)CCC4)=O)C2)=O)cnc1C(F)F CN1CC(C)(C)CC1C(=O)NC1CC(CCNC(=O)CCC2CC2(Cl)Cl)C1 c1(NCC2N(Cc3c(OC)ccc(C)c3)CC2)ncnc2ccc(I)cc12 C1(C(N(C)CCc2cccc(C#N)c2)=O)CCCCC1(C)C C12(NCCC3CCN(C(CNC(=O)C=Cc4ccco4)=O)CC3)CCC(CC1O)C2 C1(CCNC(Cc2cn(CC)nn2)=O)CCCN(C(=O)CCCCSC)C1 c1(CN(C)Cc2ccc(OC)cc2)ccc(OC)c(-c2conc2C)c1 N1(C(C=C(C)C(C)(C)C)=O)CCC(CNC(C2(C)CCC(=O)O2)=O)C(CO)C1 N1(C(C2CC(C3CC3)=NO2)=O)CCCCC(C2CN(C(C3CC34CCC4)=O)C2)C1 CC1CCc2[nH]c(=NCc3nncs3)[nH]c(=NCCCCN3CCCCCC3)c2C1 C1(CNC(CSc2c(C)n[nH]c2C)=O)CN(C(=O)C=CCO)CCC1(F)F.CN c1(CC(N2CC(CNC(c3coc(C(F)F)c3)=O)C2)=O)csc2ccccc12 C1(C(N2CCC(CSC)C2)=O)CCN(C(C2CC(=O)C2(C)C)=O)CC1 N1(C(Cc2c(C)con2)=O)CCN(C(=O)CCc2c(C)noc2C)C(CO)C1 c1(OC)ccnc(C(N2CCC2CNC(c2cncc(C(C)C)c2)=O)=O)c1OC c1(OCCCNC)ccccc1NC(c1scnc1I)=O C1(NC(C2C(COC)C2)=O)CC12CCN(C(c1cnn3c1OCC3)=O)C2 N1(C(=O)OCC)CCC(N2CCNS2(=O)=O)CC1.C12(CCOC1)C(=O)OC2 CCCCCC(CC)C(=O)N1CCCC(F)(CNC(c2cnn(C)c2C)=O)C1 C1(CCNC(c2n(CCCSC)nnn2)c2csc(Br)c2)CCC(F)(F)C1 c1(OCC(=O)NCCC(C)NC(C(CC)n2ccnc2)=O)ccccc1C(C)C c1(CC(=O)N(CC(C)NC(C2(CCCC)CC2)=O)C)ccnc(OC)c1 N1(C(CC2(C=C)CCC2)=O)CCCN(C(=O)Cc2nn(C)cc2Cl)C(C)C1 c1(CNCC2(C)CCCC2O)cc2c(nn1)CCC2 c1(C(N2CC3(CN(C(Cc4c(C)n(C)cn4)=O)C3)C2)=O)c(F)ccc(F)c1F c1(C(=O)NC2CC(C)N(C(=O)Cn3cc(N)cn3)CC2)coc2ccccc12 CC(C)(CC(=O)NCC(CC(F)(F)F)NC(=O)C1CCc2nccn21)C(F)(F)F N1(C(c2c(C)onc2)=O)CCC(C)C(NC(c2cc3sccc3s2)=O)C1C c1(CC(=O)NC(CCCNC(C2(CCC)COC2)=O)C)ccccc1C CN1CCN(C(c2ccoc2)=O)C(CNC(C2(Cc3ccccc3F)CC2)=O)C1 O(NC(=O)CC(C(F)(F)F)NC(=O)C(CC(CC)CC)CC)CC1CC(=C)C1 N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(c2cc3sccc3cn2)=O)CC2(CC2)C1 Cc1nn(C)c(F)c1C(=O)NCC1(C)CCC(NC(C23CC(CCO2)C3)=O)C1 C1(NC(C#CCNC(C2CC(=O)NC2)=O)=O)CCC(=O)NC1 c1(CC(=O)N(C(CCNC(COCCCOC)=O)C)C)ccnc(F)c1 N1(CC)CCOC(C(N2CCC(C)C2CNC(c2cccn2C(C)C)=O)=O)C1 c1(C(N2C(CNC(C3CSCC(=O)N3)=O)CC(OC)C2)=O)coc2c1COC2 c1(C(=O)NCC#CCNC(C(C)NC2CC2)=O)ccc(S(=O)(=O)N2CCCC2)o1 C=CCCCC(C(=O)NC(CO)CCOC)NC(c1ccc[n+]([O-])c1)=O C1(C(=O)NCCOCCOCCNC(=O)Cc2cncs2)COCC2(CCC2)O1 N1(C(C(CC)NCC)=O)CCC(C)(CNC(c2sc(COC)nc2C)=O)C1 c1(C(=O)NC(C(=O)NC(CC=C)CC)Cn2cccn2)ccnnc1C C1(NC(C2C(C)C2)=O)CN(C(=O)CCc2cccc(O)c2)C(C)(C)C1 N1(C(CCC=C=C)=O)CCN(C(=O)CC2CCSCC2)C(CCCC)C1 CC(CCO)C(=O)NCC(C1CCN(C(=O)CN(C)Cc2ccccc2)CC1)O c1(CN2CCC(C(=O)NCC(F)F)C(O)C2)ccc([N+](=O)[O-])cn1 C(=O)(CCC(F)(F)F)N(CC(=O)NCCC1CC1C1CC1)CC#C N1(C(CCC(C)OC)=O)CC2CC1CN(C(=O)CCN1CCC(O)C1)C2 N1(C(c2ccc(C(C)C)s2)=O)CCN(C(=O)CC2CCC(C)C2)C(C)C1 N#Cc1cc([N+](=O)[O-])ccc1COC(=O)CC(C(F)F)c1ccc(F)cc1 C1(CNC(c2n(CCC)ccc2)=O)CCN(C(c2nnsc2C(F)F)=O)C12CC2 C1(C(=O)NCC(c2ccccc2)O)CN(C(c2ccc(Cl)cc2)=O)CCC1O c1(CC)ccc(C(=O)NCc2ccc(C(=O)NC3CC(CO)C3(C)C)s2)cc1.SC N1(C(CCC)C)CC(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1=O CC1C(NC(=O)C2=COCCC2)CC2CCC1N2C(=O)CCCc1cnn[nH]1 CN1CCC2C(CCCN2S(=O)(=O)c2cccnc2NCCCCCCC2CC2)C1 CCC(CC)(CC)C(=O)NC1CC(NC(C2CC(O)CN2C(C)=O)=O)C(O)C1 N1(C(C(CC)SC)=O)CCCN(C(c2cc(C)c(Cl)s2)=O)CC1C(C)C c1(C(=O)NC23CC(C(N4CCC(F)(F)C(F)C4)=O)(C2)C3)ccc(Cl)c(Cl)c1Cl c1(OC)ccc2cc(C(N3CC4(CNC(=O)COC)CCC3CC4)=O)nnc2c1 c1(OC)cnc(Cl)c(C(=O)Nc2ccc(NC(=O)CC3CCCC3C)c(F)c2)c1 c1(C(C(=O)NC2(CO)CN(C(C3N(C(C)=O)CSC3)=O)C2)C)c(C)nn(C)c1C c1(C(=O)NC(CN(C(C2=C(C)OCC2)=O)C)C)nnn2c1CCCCC2 C1(NC)CCN(C(C)(C)C)C1=O.C1(OC)CC1N(C)C.N(C)C N1(C(C(=O)N(CC)Cc2ccc(O)cc2)=O)CCCCC1C c1(OC)ccc(C)c(C(C)NCC2(c3ccc(F)cc3)CCCCC2)c1 CC1=C(C(=O)N(C(C)(C(=O)Nc2cncc(C3CC3)c2)C2CC2)C)CC1 C1(NC(CCCOCCOCCOC)=O)CN(C(=O)CN2CCCC2)C2CC12 N1(C(C(C2CC2)OC)=O)CC(C(=O)Nc2cc(F)ccc2C)C2(CCC2)C1 C1(C(=O)NCCC(C)N(C(c2cnc(OC)c(C)c2)=O)C)CC2(C1)CC(C)(C)C2 C(=O)(C1OCCc2ccccc21)NCC1C(C)(C)CN(C(c2cnco2)=O)C1 CCC(C)(C)CCNC(=O)C(Cc1ccco1)NC(=O)CC1CNC(=O)O1 C1(CC(=O)N(CC(C)C#N)C)CN(C(C2CNC(=O)N2)=O)C(C)(C)C1 C(=O)(C(CNC(c1ncnc(C)c1C)=O)C(C)(C)C)NC1(CC(=O)OC)CC1 Cc1cnc(C(=O)N(C)CC2CCN(C(c3ccc(C(C)F)cc3)=O)C2)nc1 c1(C(=O)OC(C)C(C)(C)C)ncccc1CNC(=O)OC(C)(C)C N12CCN(C3(CCCOC3)C1)C2=O.CCCCCCc1ccc(C(C)OC)cc1 C(C(C)CC(=O)NCCCCCC1CC1)NC(C1(COC)CC(=O)C1)=O CC1CN(C(C2CC3(CCC3O)C2)=O)CCC1C(=O)N(CC(=O)N(C)C)C c1(C(=O)NCC(=O)NCC=C)sc(-c2ccccc2Cl)nc1C N1(C(C2CCC(CNC(c3n[nH]c(=N)[nH]3)=O)O2)=O)Cc2c[nH]nc2C1 Cc1ccc(CNC2CCN(S(=O)(=O)c3cn[nH]c3)C2)cc1O C1(CNC(CC=C)=O)CN(C(=O)COC2CCC(C)CC2)CC1C C1(C(=O)NCCN(C(c2cc(C3CC3)ns2)=O)C(C)C)(OC)CC(C)C1 Cc1cccc2c(CCC(N3CCC(CCNC(C4CC4F)=O)C3)=O)c[nH]c12 N1(C(C(C)OCCOC)=O)CCCC(C)(C)C1C(=O)N(CCO)CC1CC1 c1(C(N(CCCNC(C2CCSCC2)=O)CC)=O)ccn(C(C)C)c1C c1(NC)ccc(CNC(c2ccccc2C(=O)O)=O)cc1F C1(CNC(C(CC)C)=O)CC2CCC(C1)N2C(=O)CCc1cncn1C N1(C(COCCC(C)C)=O)CCC(C)(NC(C2CC3(CC3)CO2)=O)C1 c1(OC)ccc(Cl)c(CC(=O)NC2CC(C)N(C(c3cn(C)cn3)=O)C2)c1 N1(C(c2ccn(C)n2)=O)CC2CC1(C(=O)NCCCSC(F)F)C2 c1(COCC)cccc(CNC(=O)Nc2ccc(N3CCCC3)nn2)c1C c1(CC)ccc(C(=O)NCC2CN(C(C3CCCCS3)=O)CC2C)cc1 N1(C(C2CCN(C(=O)NC(CCC)C)CC2)=O)CCC2(C1)NC(=O)N(C)C2=O CCC(CNC(C1CC(C)CN(C(=O)CCCOC(C)C)C1)=O)C(C)(F)F C(=O)(C(F)C(C)C(F)(F)F)NCCCNC(C(n1cc(C2OCCO2)nn1)C)=O c1(C(C(=O)NCC(C)(C)NC(=O)C(C)N2CCCC2)SC)ccccc1 n1(CC)ccc(C(N2CC3CC(C2)C3NC(=O)CC(O)C(C)C)=O)cc1=O N1(c2nc(C)c(Br)cn2)CCC2(CCN(C(=O)C(C)(C)CO)C2)C1 n1(CC(=O)OCCOCCOCc2cscn2)c(-c2cccs2)nnc1S N1(C(c2ncc(C)cn2)=O)CCC2(CCCN(C(=O)CC3CSC3)C2)CC1 n1(CC)ncc(C(=O)NC2COCCC2NC(=O)CN2CC(C)C2)c1Br Cc1cc(C(N2CCC(CNC(C3CCOC3)=O)CC2)=O)nn1CCO c1(C(=O)NC(C(C)C)CCNC(C2CCCC23CC3)=O)cccc2c1OCC2 c1(C(N2CCC(CN(C(CCC(=C)Cl)=O)C)C2)=O)nccc(N)c1Cl c1(C(N(CC(C)NC(c2cc(C)nn2C)=O)C)=O)ccc(Cl)c(F)c1F N1(C(CCC(C)(C)C(=O)OC(C)(C)C)=O)C2CCCC(O)C1CC2 c1(C(=O)NC2C(NC(C(C)Oc3ccccc3Cl)=O)CC2)nc2ccccc2o1 c1(N2CCC(CC=C)(NC(C3CCCC3CC)=O)C2)ncnc(Cl)c1CO C12(C(=O)NC(CCC)CCC)CCC(CC1NC(=O)C(CC1CC1)OC)C2 C1(CNC(C(CC=C)OC)=O)CC(C(=O)NC(C)CCN(C)C)=NO1 N1(Cc2c(O)ccc(C#N)c2)C(C(=O)Nc2cccc(O)c2)CC2CCCCC12 c1(CC(C)C(=O)NC2(C(=O)NC3CC(F)C3)CC2)cccc(C(F)(F)F)c1 N1(C(CC(CC)C2CC2)=O)CCC2(CCC(NC(=O)CCCCOC)CC2)C1 C=C(C)C1OCCC1C(N1CC(C(O)C(=O)NCC(N2CCCC2=O)C)C1)=O CCCCC(CNC(c1cccc(Cl)c1)(C)C)CC C(C(C(C)C(C)C)NC(=O)C=CC1CCC1)NC(c1ccc(OCCC)cc1)=O N1(C(C2CC(C#C)(O)C2)=O)CC2(CC(C(=O)NCc3nnnn3C)CO2)C1 C12(NC(c3n(CCC)ccc3)=O)CCC(CC1)N(C(c1ccc(CSC)o1)=O)C2 C1(NC(c2c[nH]c3nccc-3c2)=O)CC2CC1CN(C(c1ncc[nH]c1=O)=O)C2 c1(CN2CC3C(C(=O)NCc4ccc(C)nc4)(C3)C2)[nH]nc2ncccc12 CC1(C)C(C(F)(F)F)CCS1(=O)=NC=O.CN CCC(C#N)C(=O)N1CC(CC(C)NC(c2occc2COC)=O)C1 C1(CC)CN(C(=O)C(C)(C)c2ccno2)CCN1C(C1(C2CCCS2)CC1)=O c1(OC)cccc(C(=O)NC(C)CCNC(=O)C=Cc2ccc(C(N)=O)o2)c1 O=C(CC(O)CNC(c1ccc[n+]([O-])c1)=O)Nc1ccccc1C1CC1 C1(C(=O)NC(C(=O)NCCOCCOC)c2ccoc2)CCCN(C)C1 CC(=O)CCCCC(=O)N1CCC2CN(C(=O)C(C(C)(C)C)n3cnnn3)CC12 C1(CC(=O)NC(CNC(C=CCN(C)CC)=O)CO)CC2C=CC1C2 Cc1ccc(NC(C2CC(O)CN2C(c2ncc[nH]2)=O)=O)c(CN(C)C)c1 c1(N2CC3CC(NC(=O)C=CI)C3C2)ncc(Cl)cc1[N+](=O)[O-] N1(C(C=CC)=O)CC(NC(c2cc(Br)c(Cl)s2)=O)CC(F)(F)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(=O)CCc2ccnn2C)CC(O)C1 Cn1nnc(C(N2CCC(C(C)(C)C(=O)NCCc3cocn3)C2)=O)c1N CC1CC=C(C(=O)NCC2(CNC(c3cccn4nnnc34)=O)CC2)CC1 CC(C(=O)NNC(=O)c1cccc2c1OCC2)NCc1ccoc1 C1(CC=C)(NC(=O)CC2CC(C)N(C(c3cnc(C)nc3)=O)C2)CCOCC1 N1(CC)CCCC(C2CCN(C(C3(C4(O)CCOCC4)CC3)=O)C2)C1 C1(CNC(c2c(C)scn2)=O)CCN(C(=O)C=CC2COC(C)(C)O2)CC1(F)F CC1CN(C(=O)CN(C2CC(C#N)C2)C(c2cccc3cc[nH]c23)=O)CC(C)(C)C1 C(=O)(C(CC1CCC1)[N+](C(=O)C=CCc1ccsn1)([O-])CC)NCCOCC=C CC1=C(C(=O)NCC=CC(=O)N(C2CCO2)CC2CC2)CC1 c1(C(=O)NC2C3N(C(c4c(NC)cnnc4)=O)C(CC3)C2)ccc(F)c(F)c1F C1(C(N(CC(O)CO)C)=O)(NC(C2(C3(C)OCCO3)CC2)=O)CCSC1 S(=O)(=O)(c1cnn(C)c1)N1CC(CC(=O)Nc2c(OC)cc(F)cc2)C1 Cc1cc(C(=O)NC2CN(C(C3CCCC3)=O)CC2O)c2cnccc2c1 C(=O)(C1=COCC1)N(CC(CC)NC(c1nc(Cl)cs1)=O)CC c1(-n2cc(CCC(=O)N(C(C(=O)OCC)C)C3CC3)nn2)ccc(Cl)cc1F CN1CCN(CC(=O)NCC=C2CCN(C(=O)C(c3ccc(Cl)s3)=O)CC2)CC1 N1(C(C2CC(SC)C2)=O)CC2CC(C(=O)NCCc3cccc(F)c3)(C2)C1 N#Cc1c[nH]c(C(=O)NCC(=O)NCCn2ncccc2=O)c1 Cc1nn(CC(N2CCC2c2cn(C3CCCOC3C(C)C)nn2)=O)c(C)c1C n1(COc2ccc(OC)cc2)ncc2ccccc12.c12ccccc1O2 c1(NC(=O)CCOc2cccc(Br)c2)ncn2cc(C(N3CC4CC4C3)=O)sc12 c1(C(=O)NC(CC(N2C(COCC)CCCC2)=O)C)ccc(C#N)cc1 C1(C(N(CCCN(C)C)CCC)=O)(CC)CCCN(C(c2cccc(C#N)c2)=O)C1 C(=O)(C=CSc1nc[nH]n1)N(CCNC(c1cnc(CO)s1)=O)CCOCCO c1(C(=O)NC(CCCCNC(C(CO)OC)=O)(C)C)cc(C)cc(C)c1C C(C)(C(C(=O)NCCN(C(C1(c2ccccc2)CC(O)C1)=O)C1CC1)N(C)C)OC N1(CCC)C(=O)CCC1C(=O)NC1(CF)CCN(C(=O)Cc2cncc(O)c2)C1 n1(CC)nnc2c1C(C(=O)N1CC(OC(C)(C)C)C1)CN(C(=O)CCc1ccncc1)C2 c1(NC(Cn2cc(CC)nn2)=O)cc(C#N)cnc1C N1(C(CC(C)(F)F)=O)CCOCC(CNC(C23CCCCC2C3)=O)C1 CC(CN=C(NC(C1CC1)C1CC1)NCC(C)(Cc1ccccc1)C(N)=O)CC(F)(F)F N1(C(=O)OC)CCCC2C1CCCN2C(c1ccc(C(=O)OC)s1)=O c1(CN2CC(C)(C(=O)NC(COC)C3CC3)C2)ccc(-n2cccn2)nc1 N1(C(c2noc(C)c2Br)=O)CCC2(CCCN2C(C23CCCC2C3)=O)CC1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(c1coc(-c2ccccc2)n1)=O c1(C(=O)NCC(CC)(C)NC(C2CCCC(OC)O2)=O)cnn2ccnc(C)c12 N1(C(C2C(SC)CCC2)=O)CC2CC(C1)C2NC(C1CC2CC2C1)=O c1(C(=O)NCCN(C2CCC(C)CC2)C(C(C)SCC)=O)ccc(F)cc1F C(CCCCCn1ccnn1)N(C)C(=O)OC(C)(C)C.C1C(O)CN1 CCC(C#N)C(=O)NCC1CN(C(C2CC(=O)N(c3ccccc3F)C2)=O)C1 c1(C(=O)NCC(C(C)C)NC(C(C)SC(F)(F)F)=O)ccc(N)c(Cl)c1 N1(C(C(C)OCC#C)=O)C2CCC1CC(N(C(=O)C(F)(F)CCCC)C)C2 C#Cc1cccc(C(=O)NC2CC(O)CN(C(=O)CCC3CCCC3)C2)c1F c1(C(=O)NC(C(C)NC(C2(COC)CC=CC2)=O)C)cc(OC(F)F)n(C)n1 N12CCC3(CC1)CC3C2=O.N#CC1CC(NC(=O)CCc2cncnc2)C1 CCCC(C)CCNC(=O)CNC(=O)CNC(c1c[nH]c(=N)o1)=O C1(NC(Cc2cc(C)no2)=O)CN(C(c2ccc(N3CCC3)cc2)=O)CC2CC12 n1(C(C)C)ccnc1C(=O)NCc1ccc(C(=O)NCC2CCC(O)C2)s1 c1(NC(C(C)(N(C(CC=CCC)=O)C)C2CC2)=O)ccn2nccc2c1 CCCC(CNC(C1(OC)CCCC1)=O)C(=O)N(CCCO)OC Cc1cc(I)ccc1C(C)Nc1cc(NCc2ncc(Cl)n2C)ncn1 c1(C(=O)NCCNC(C=C2CCN(C)C2)=O)nc(Br)[nH]c1C(F)(F)F N1(C(c2ccc(C)cc2)=O)CCC(NC(C2CC(C(C)C)C2)=O)C(O)C1 CCCC(C)(CCC)C(=O)N1CC(CNC(c2[nH]nnc2C)=O)C(C)(C)C1 N1(C(C2(C)CCCCC2)=O)CCC(N=c2ccnc(Cl)[nH]2)C(F)(F)CC1 c1(CC)ccc(C(=O)NCCOCCCNC(C2CCCC(C)CC2)=O)cc1N O=C(C1CCc2cccnc21)N1CC2CCC(C1)N2C(c1cncs1)=O c1(C(=O)N(CCCC)OC(c2ccc(CN3CCCC3)o2)=O)nc(C)ccc1F C1(C(=O)OC)CC=CCN1C(c1ccc(CO)o1)=O.C12CCC(CC1)CNC2=O C(C)(C)(CCNC(=O)C=CSC)NC(C1(COC)COC1)=O c1(OC)ccc(F)cc1C(=O)NC1CC1CNC(c1cc(C)n(C2CC2)c1C)=O C12(C(=O)NCC3CCCCN(C(C(C)SC(C)C)=O)C3)CCCCC(F)(C1)C2 c1(NC(CC)(CNC(C2COC(C)C2)=O)CC)nc(C)nc(=N)[nH]1 c1(C(=O)NCCCN(C)C(c2cnn(C)c2)=O)cccc(S(C)=O)c1 C(=O)(C(F)CCC(C)C)NCC(CC(=O)N(C(CC)(C)C)CCO)OCC c1(C(=O)NCC(CO)NC(=O)COCC2CCCOC2)c(O)nnc2c1CCC2 C(=O)(C(O)CCCCC)NC(C(=O)NC(CC=C)(C)C(F)F)C CC(CC(C)NC(c1cc(F)c(F)cc1F)=O)N=c1[nH]nc(CO)s1 Cn1nc(C2CCCN2C(c2cc3cc(Br)cn3cn2)=O)c2ccccc2c1=O c1(C(=O)NCC(Cc2ccccc2)N(C(C2C(C)C2C)=O)C)cn(C)c(=O)cn1 c1(C(=O)NCC(CNC(C2CCC(C(=O)OC)C2)=O)O)nccn2cc(C)nc12 N1(C(C2C(CCOC)C2)=O)CC(NC(c2cnc[nH]2)=O)C(SC)C1 CCC(C(=O)NC(C)(CNC(c1c(OC)ccc(Cl)c1F)=O)C(C)C)C(F)(F)F O=C(CCC(=O)N1CCC(O)CC1)NCC1CC1CNC(c1ccc(Cl)[nH]1)=O C1(C#N)(C(N(CCOCCN(C)C(c2cncs2)=O)C)=O)CCCCC1 C(CCC(=O)NCCNC(=O)CCCC1CC1C)NC(C)=O.C12CC1CNC2=O N1(CC(=O)NCc2ccco2)CC2CC(NC(c3cccs3)=O)C1C2.C(=O)(C1CC1)N C1(CNC(C(C=CC)O)=O)CN(C(C2CC2c2ccccc2)=O)CC12CCC2 C#CCC(C(=O)NCC1CCN1C(C)(C)C)NC(c1cnn(C)c1Cl)=O c1(C(=O)NCCCNC(c2c(C(C)(C)C)nc(C)s2)=O)cnn2cccnc12 N1(CC=C)C(=O)CCN(CC(N2CCCCC2)=O)C1=O.C=CCN(CCSC)C C(=O)(C1=CCCCO1)NCc1ccc(C(N2C(C(CCC)C)CCC2)=O)s1 Cc1ccncc1CC(=O)NCCC1CN(C(=O)C(C#N)=CC(C)C)CCO1 C#CCC(O)C(=O)N1CCC(CNC(c2cccc(-c3cccc(C)c3)c2)=O)C1 c1(NC2CN(C(c3cnc(C)o3)=O)CC2C)ncc([N+](=O)[O-])cc1Br c1(OCCOC)cccc(NC(=O)C(N2CCOC(COC)C2)c2cc[nH]n2)c1 c1(C(c2n(CCSC)nnn2)NCC(C)OC(C)(C)C)cccc(C)c1F C1(NC(C2(CC)CC2(F)F)=O)CCN(C(C2CSCN2C(C)=O)=O)CCC1CO C1(CN(C)C(C2(C(N)=O)CC2)=O)CCN(C(c2cc(Br)ccn2)=O)CC1 O=S1(=O)CC2CC1CN2C(=NCc1cccc(O)c1F)NC1CCC1 N1(C(c2nncc(OC)c2)=O)CCCC1C1CCCN1C(c1cccnn1)=O Cc1ccc2c(C(N3CC(F)(F)CC3CCNC(=O)CCC(N)=O)=O)onc2c1 c1(C(C(=O)NCC2CC(=C3CC3)C2)N(C)C(C2CC2(F)Cl)=O)ccnn1C C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)C#CC2CC2)CC1C(F)(F)F N1(C(C2C(c3cn(C)nc3)C2)=O)CC2CC(C1)CN(C(c1[nH]ccc1C1CC1)=O)C2 N1(C(CCCC2C(C)C2)=O)CCCN(C(C23CC(C(=O)N(C)C)(C2)C3)=O)C(C)C1 c1(C(C(=O)NC2COC2)N(C2COCCN(C)C2)C)nn(C)c2c1CCC2 c1(C(N(CCCNC(=O)C(c2cccs2)SC)CC)=O)nccc(Cl)c1C C1(O)(CCNC(C2CCCCCCC2)=O)CCN(C(C2CCCC(F)C2)=O)CC1 C(C(CC(C)C)C(=O)NC1COC(C)C1)OC C1(C)(C(=O)NCCCNC(C(Cc2ccc(C)cc2)C)=O)CC(C(C)(C)C)=NO1 c1(-c2nc(NCc3ccc(OCC(C)C)nc3)sc2)cc(Cl)ccc1OC(C)C c1(OC)cc(Cl)c(C)cc1NC(=O)NC1CC(c2cccc(F)c2)(F)C1 CCC(CCOC)C(=O)NC1COCC1NC(c1cc(O)n(CC)n1)=O ClC=CCN=c1[nH]c2c(c(=NC3CN(CC4CCOCC4)C3)[nH]1)COCC2 C(C(CO)(CO)NC(C1CC1F)=O)N(C(c1ccn(CC)n1)=O)C n1(CC)nnc2c1C(C(=O)N1CC3OCC(C)C3C1)CN(C(=O)C(C)COC)C2 N1(C(CCC=CC)=O)CC(NC(=O)CNC(=O)NC)CC2(CC2)C1 c1(CC)nc(Cl)c(F)c(=NC(CNC(=O)CCSC)CC)[nH]1 C12(NC(=O)NC3(c4ccc(F)c(F)c4)CCC3)CCCCCC1OCC2 N1(C(c2cccc(NC)n2)=O)CC2CN(C(=O)C(c3cccnc3)C)CC2C1 c1(C(=O)Nc2c(C#N)cccc2)cnn2ccc(-c3c(F)cc(F)cc3F)cc12 C1(Cl)(C(N(C)CC2N(C(c3ccn(CCN(C)C)n3)=O)CCC2)=O)CC12CCC2 c1(NC(C2CN(C(C3C(C=C)C3)=O)C2)=O)ccccc1CCN(C)C C1(C(=O)NCCCC2N(C(C(c3n(C)ccc3)=O)=O)CCC2)CC(F)C(=O)N1 c1(N2CCCC(SC)C2)nc(NCC(F)(F)Cl)nc2c1CCCC2 c1(CNCC(CNC(CCC(=O)c2cn(C)nc2)=O)(C)O)c(Cl)ccc2c[nH]nc12 N1(C(=O)NC23CCC(Sc4ncccn4)(CC2)C3)CCc2c(F)cccc2C1 N1(C(CC(C)OC)=O)CC(CNC(=O)CSc2cccc(C)c2)C(C)(C)C1 c1(C(=O)NC(C)CCNC(=O)Cc2ccccc2Cl)ccc(-n2cccn2)cc1 n1(CCC(=O)NC2C(CNC(=O)CCC(F)(F)F)CC2)cc([N+](=O)[O-])cn1 c1(C(N2CC(N(C(C)=O)C)C(F)C2)=O)n[nH]c2cccnc12 C1(C(N2CC(CN3CCN(C(=O)CCF)CC3)C2)=O)COc2ccc(F)cc2C1 C(=O)(CC1NC(=O)c2ccccc21)N(C)CC1CCCN1C(=O)C=CCF c1(C(=O)NCCN2CCN(C(CC3C(C)C3)=O)CC2)c[nH]c2cc(F)c(F)cc12 O(N(CC)C(=O)CC1CCC(NC(=O)COc2cccc(O)c2)C1)CC Cc1csc2cc(C(N3CC(NC(=O)CCC4(C)CC4)C4CC4C3)=O)[nH]c12 C1(C(N(C)CCC2CCCCC2)=O)COCCN(C(C2CC(C3CC3)=NO2)=O)C1 N=c1ccc(C(=O)NC(C(=O)NCCN2CCCOCC2)C2CCCO2)c[nH]1 N1(C(C(CO)NC(C(=O)OCC)C)=O)CCC(C(=O)Oc2ccccc2)CC1 C(=O)(C1=CCCC1(C)C)NCCCN(C(C)C)C(C1Cc2nccnc2C1)=O CC(C)C(C)C(=O)NC1CCCC(NC(c2cocn2)=O)C1 CN1CCN(CCCNC(=O)N(CCO)Cc2ccc(Cl)cc2)CC1 CCCC(CCC)CC(=O)N1CCC(C(=O)NCCCNS(C)(=O)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC1C(C)(NC(=O)CSC2CC2)CCCC1 c1(C(N2CC(OCC)C2)=O)ccc2c(n1)CN(C(c1cnncc1C)=O)CC2 C1(C(N2CC(C)C(CNC(=O)CN3CCSCC3)C2)=O)CCCC(C)(C)C1 C(=O)(C(C)C(O)CC(C)C)NCC1(O)CCCN(C(c2c(C)c(Cl)cnc2)=O)C1 c1(Nc2cc(OCC)ncn2)ccc2c3c(cccc13)CC2 c1(-c2cccc(OC)c2F)ccc(S(=O)(=O)N2C(CO)CCC2C)cc1 c1(-n2c(C3ON=C(C)C3)nc(-c3ccc(C4CC4)cc3)n2)cc(C)ccc1C c1(C(N2C(C)CN(C)CC2)=O)cc(O)nc2c1CN(C(=O)CSCC(N)=O)CC2 c1(C(=O)NCC(C)(O)Cn2cc(Br)cn2)cc(C2CCC2)cnc1O CCCCC(F)C(=O)NC1CC2CC(NC(c3cccc(C)c3Cl)=O)C1C2 N1(C(C(=O)NC(C)C)=O)CCC(C)C(NC(c2coc(C(N)=O)c2)=O)C1C C1(OC)CN(C(c2cc(-c3cnn(C)c3)[nH]n2)=O)CC1NC(=O)C(C)(C)F CCCCCC(O)CC(=O)N1CC2CCCC2(NC(C2CNC(=O)N2)=O)C1 Cc1[nH]c(C(=O)N(CC#N)CC#N)c(C)c1C(=O)Nc1nc(Cl)cnc1Br C1(C(N2CC(OC)(CNC(=O)CN3CC(C)C3)C2)=O)CCC(=C(F)F)CC1 c1(COC)nc(C(=O)N(C(C)C(=O)NCC2(F)CCC2)C)co1 c1(OC)ccc(CCCC(N2CCOC(c3ccc(Br)cc3)C2)=O)c(Cl)c1 c1(NC(C2CCC(C)N2C(=O)C2=CCCCO2)=O)cccc2cccc(Br)c12 Cc1ccnc(CC(=O)NC2CCC2CNC(c2cnc(O)n2C)=O)n1 Cc1ccc(NC(C2(C)CCN(C(=O)Cn3cc(Br)cn3)C2)=O)c(Br)n1 C(CCC(C(=O)NCCC1CN(C)C1)NC(c1cnco1)=O)OC c1(NC)cnccc1C(=O)NCc1occc1C(N1CCCC1CO)=O CC(C)C(F)C(=O)N1CCC(C(C)CNC(C2CN(C3CCOCC3)C2)=O)CC1 C1(O)(C(C)NC(C2CC3CCCC23)=O)CCN(C(=O)CCC2(C)CC2)CC1 c1(C(N2C(C)CC(NC(c3cnco3)=O)CC2)=O)cc2ccc(Br)cc2s1 c1(C(=O)NC(CNC(C(F)=CC)=O)(C)C2CCC2)ccnc2c(F)cccc12 Cc1nn(C)cc1C(N1CCC1CNC(=O)C(c1ccc(Br)cc1)C)=O CCC(CC(=O)N1CCOC(C(N)=O)C1)N(C)C(C1CC1C(F)F)=O C1(C(=O)NC(C=CC(=O)NCC2(CC=C)CCCC2)C)CCCN(C)C1 C12(NC(CC3(C)CCN(C(=O)C=Cc4ccsc4)C3)=O)CCCC(C1)OC2 C=CCN=C(NCc1ccc(F)cc1C)NCC1CC(C)(c2ccccc2)C1 CCCC(CC)CCC(=O)NC(CN(C)C)C(=O)NCC(C)(C)C(N)=O C1(CNC(CCc2cn(C)nn2)=O)CCN(C(c2cccc(O)c2Cl)=O)C12CC2 N1(C(c2cccc(OCc3ccccn3)c2)=O)CCC2(CCC(O)C2)CC1 S(=O)(=O)(c1cnc(N2CC(C3CC3)OC(C)C2)c(Cl)c1)NCc1ccc(CC)s1 N1(C(C2(C)CCNC2=O)=O)CCCC2(C1)CN(C(C1CCCCS1)=O)C2 c1(NCCNC(C2(c3cccc(F)c3)CC2)=O)c([N+](=O)[O-])cccc1[N+](=O)[O-] N1(C(c2c(C)occ2)=O)CC(C(=O)NCCN=[N+]=[N-])C(C)C1 C(c1ccc(F)cc1)=C(C(=O)N(C)CC1CCN(C(C(C)NC(=O)NC)=O)C1)C c1(CNC(CN(C)C(c2cccc(C=O)c2)=O)=O)cnc2ccccc2c1.C(=O)O C1(=O)C(C)(C2CC2)N1.C(C(=O)NC)SCC.C1(=O)CN1CC N1(C(C23CC(NC(C(C)NC(=O)C4CC4)=O)(C2)C3)=O)CCCC(C)C1C C1(N(C(c2cccc(C)c2)=O)C(c2ccc(F)cc2)C)CCC12CCNCC2 C(=O)(CCCC(=O)NC1CC(C)N(C(=O)CCCn2cccn2)C1)NCC N1(C(C=CC=CCC)=O)CC(F)CC1CNC(=O)Cn1nnc(C)n1 C1(C(=O)NCC(C)(C)NC(C2(C(F)(F)F)CCCC2)=O)CC=CCC1 c1(C(N2CCCC(CNC(CC3(N(C)C)CCC3)=O)C2)=O)cnc2ccoc2c1 C1(C(N2C(C)CC(NC(=O)CC3OCCC3(C)C)C2)=O)CCC2(CCC2)O1 N1(C(C2OCCN(C)C2)=O)CC(CNC(C2(O)CCC2)=O)C(F)(F)C1 C1(C(N2C(C)(CNC(c3cccc(N)c3)=O)CCC2)=O)CCCCC1(C)C c1(Nc2ccc(C(=O)NCC)cc2)cccc2ccoc12.C12CCN1NC2=O N1(C(CC(C)(C)OC)=O)CC2(C(=O)N(C(C)C(C)C)C)CCC1CC2 C(C(C)(O)CC(=O)NCCCNC(=O)C=CCN1CCCC1)OC N1(C(CSCCC=C)=O)CCC(N(C(=O)CCc2cccc(OC)n2)C2CC2)CC1 c1(C(=O)OC)cnc(C(=O)NC2CC(CCNC(C3(C)C=CCCC3)=O)C2)cn1 C(=O)(C1=C2CCCN=C2NN1)NC(C1CCCN1C(C1CC2CCC12)=O)(C)C c1(SCC(=C)C)ccc(-c2nnc(CN3CCCC(C)C3)n2N)cc1 n1(C(C(=O)C(COC2C(c3ccccc3Cl)(C)CC2)=O)O)cc(S(C)(=O)=O)cn1.OC C1(C(=O)NCCN(C(CC=CC=C)=O)CC2CC2)OCCC1C(F)(F)F c1(OC)ccc2c(C(=O)NCC(CNC(=O)CCCCC(N)=O)CO)n[nH]c2c1 C1(CN)CCN(CCNCC2(CO)CC(C)(C)C2)CC1 C1(C(=O)OC)CN(C(C2CC2CNC(C2CCC2C)=O)=O)C(C)(C)C1 C=C=CC(C)C(=O)NCC1CN(C(=O)CCc2ccn(C)n2)CC1C(F)(F)F c1(CN2CCN(CCC(=O)OC)CC2)cnc(OC)c(C)c1.C12CCCCN1C2=O CC(C(=O)NCC1(F)CC(NC(=O)C(N2CCN(C)CC2)C)C1)C(F)F c1(C(=O)NCC(CC(=O)NC2CC(OC)C2)OC)cnc(O)c(F)c1 C1(NC(CNC(=O)OCC)=O)CN(C(c2cn(C(C)C)nn2)=O)C2(CCOC2)C1 C(=O)(CC1CCOc2ccccc21)NCC(C)NC(c1c(C)oc(Cl)n1)=O c1(-c2cc(OC)cc(Cl)c2)n[nH]c2c1CN(C(c1cccnc1C)=O)CC2 C1(NC(c2cc(C)ns2)=O)CN(C(=O)C(C)(F)c2ccon2)CC(C)(C)C1 c1(OC)ccc(CC(N2CCOC(CNC(=O)CCCC3CCC3)C2)=O)c(F)c1 C1(C(N2CC3(CN(C(c4nc(C)n(C)n4)=O)C3)C2)=O)CCc2[nH]nc(O)c2C1 C(c1ccc(Cl)cc1)=CC(=O)NCC1C2CN(C(=O)CCN3CCOCC3)CC12 C1(CCOC)CN(C(c2cscc2F)=O)CCN1C(c1cc(COC)no1)=O N1(C(CSCCC)=O)CC(NC(c2ccn(CCC)n2)=O)CC12CCOC2 N1(C(C(C)(C(C)C)OC)=O)CCN(C(=O)C=Cc2ccccc2)CC(O)C1 CS(=O)CCC(O)C(=O)NCC1(NC(c2cnc(=N)[nH]c2)=O)CCC1 N1(C(C(C)C(C)S(C)(=O)=O)=O)CC2(CCN(C(=O)CS(N)(=O)=O)CC2)CC1C n1(CCC(=O)OC)cc(N(C)C)nn1.n12cc(nn1)C2(C)C.C12CN(C1)C(=O)C2 C(CO)(C(F)(F)F)NC(CC=CCNC(CCOC)=O)=O C1(CC(=O)NC(CN(C(=O)CC2CCC2(C)C)CC)C)=CN=CC=CC=C1OC C12(CCNC(c3c(CC)nn(C)c3)=O)CCC1CN(C(=O)Cc1cncn1C)C2 N1(C(c2c(C)cc(C#N)s2)C(=O)NCC2CCCO2)CCC2CCCCC12 n1(CCC(N2C(C(=O)OC)CC(n3ccnn3)C2)=O)c(C)cccc1=O c1(C(=O)NCC(CC)(C)NC(=O)CC2CC(C)C2)cc(Br)c2nccn2c1 c1(C(=O)NC2CC(NC(c3c(C)cn(C)c3)=O)C2)nnc(O)cc1O C1(CCC)CCCC(CNN(C)C)C1.c12n[nH]cc1CNC(=O)N2 c1(NCC)ccc(C(N2CC3(C2)CN(C(=O)CC(F)F)C3)=O)cc1C(F)(F)F CC1(C)CC2N(C1)C(=O)C1CN(C1)C(=O)C2.c1(NCC(=O)NC=O)ccccn1 c1(C(=O)NCCN(C(CC)=O)CCOC2CCC2)ccc(Cl)nc1OC C1(C(N(CCOC)CCNC(=O)CC2(CO)CC2)=O)Cc2nnc(C)n2C1 C(=O)(CCCCN(C)C)NC(C1CCN(C(C2C(CCC)C2)=O)C1)C N1(C(C(C)C)=O)CCC2CN(C(=O)C=CCBr)C2C1.c1(CCC=CC(=O)N)ccccc1 C1(COC)(NC(=O)CCS(N)(=O)=O)CCN(C(=O)CS(N)(=O)=O)CC1 c1(NC(c2nc(C(=O)Nc3c(OC)cncc3)sc2)=O)cc(F)cc(C#N)c1 N1(C(C(CC)n2cncn2)=O)CCN(C(=O)CCN2CCC2)CC1CC c1(CCC(=O)NC2CCC(NC(=O)C=CC=C(Cl)Cl)CC2)nnc(O)nc1O C(=O)(C1=NOC(C)C1C)NC1(C(N2CC3C(OC)(CC3)C2)=O)CCSC1 N1(C(C2CC(NC(c3coc(Cl)n3)=O)C2)=O)CCOC2(CCS(=O)(=O)CC2)C1 CC(C)CC(CNC(C1CCC2(CC2)C1)=O)C(=O)NOCCC(C)C C(=O)(C1CCCc2nc[nH]c21)N(CCCCCNC(C1CCS(=O)(=O)C1)=O)C Cc1nc(CNc2cc(C(C)C)ccc2C)c(F)c(C)n1.N12CCCC1C2 N1(C(C(n2ncc(C)c2)C)=O)CC2CC2C1C(=O)N(CC1CC1)CC1CC1 C(C)(C)(CCCC(=O)N1CC2(COC(=O)C2)C1)NC(c1cnn(C)n1)=O c1(-c2nc(COC)nn2C2CC2)cc2c(Cc3ccc(Cl)cc3)nccc2o1 c1(C(N2C(C(C)NC(C(C)OCC)=O)CCC2)=O)cc(F)c(F)cc1O CC1=C(C)CC(C(=O)NCC(=O)NCC(O)CF)CC1 C1(NC(c2cc(COC)no2)=O)CC(CNC(c2nscc2C)=O)C(O)C1 C1(n2cc(C(CC)O)nn2)CCN(C(=O)C(c2cccc(COC)c2)(F)F)CC1 C12(C(N3C(CCNC(CCCC=C)=O)CCCC3)=O)CCCN(CC1)S2(=O)=O CCCC(C)(O)CC(=O)NCC1CCN(C(=O)CCC2CCCO2)C(C)C1 c1(C(=O)NCCCN(C(c2c(C)c(F)ccc2)=O)C2CC2)cc2c(s1)CCCC2 N1(C(C2CCN(C(C(C)C(F)F)=O)C2C)=O)CCCC2(CCC2)CC1 c1(CCC(=O)NC2(CNC(=O)Cn3cncn3)CCCC2)cccc(F)c1F C(=O)(C(=O)C(C)(C)C)NCC(CO)NC(CCCOCCC)=O c1(C(=O)NCC2CN(C(CC(C)CC(C)(C)C)=O)C2)cc(N)cc2ccccc12 c1(NC(c2nnnn2CC2CCCO2)C2(N)CC2)cccc(SC)c1.CCS C1(N(C(c2ccc(OC)cc2)=O)C)CCN(C(c2c[nH]nc2Cl)=O)CC1C c1(OC)cc(C(=O)NCCOCCNC(=O)C(C(C)C)OCOC)c(C)c(Br)c1 c1(C(=O)NCCC2(CNC(=O)CSc3cn[nH]c3)CC2)cnccc1Cl C1(C(=O)NCC(CC(=O)N2CC(CC)(CO)C2)OC)C2CC3C(C2=O)C13 c1(CSCCCNC(S(CC)(=O)=O)=O)ccccc1.C1(=O)C(=O)N(C)CC(C)N1 N1(C(C(C)C(=O)O)=O)CC2CCN(C(=O)CC(C)(C)C)CCC2C1 c1(CN2C(CC(N3CCN(CCC)CC3)=O)COCC2)cc2ccoc2cn1 Cc1nc(CN(CC2=CCCCC2)C(C)C)c(Br)[nH]1 C1(C)(CC)C=C(C(=O)N(C2CC(NC(c3cn(C4CCC4)nc3C)=O)C2)C)C1 CCCC(C(=O)NCCC1CC(C)(C)CO1)NC(=O)C#CC1CC1 CC1OC2(C)CC1(C(=O)NCCN1CCN(c3cc(C(N)=O)nc(Cl)n3)CC1)C2 c1(N2CCCC(n3c(C)cnc3)C2)c(C#N)cccc1C#N c1(C(N2CC3(CN(C(c4cc(C)n(C)n4)=O)C3)C2)=O)cn(C(C)C)c(=O)nc1O c1(OC)cc(CCC(=O)N(C)CC2(O)CN(C(=O)C(C)S(N)(=O)=O)C2)ccc1Cl C=C(Cl)CC(C(=O)NCC1(O)CCSC1)NC(c1ccc(OC)cc1)=O CC(C)C1=NOC(C(=O)NCC2CN(C(C3(C(C)C)CCC3)=O)CC2(C)C)C1 CCC(O)C(=O)N1CC(O)(C(C)NC(=O)COCc2nnc(C)s2)C1 c1(NCC(c2c(C)cccc2)C)nccc(=NC2CC(=C3CCC3)C2)[nH]1 CC1CN(C(c2ncc(C(N)=O)cc2Cl)=O)CCC1CNC(C12CC1C2)=O C(=O)(C(C)(C)CCCF)NC12C(CN(C(C(CCC)NC(C)=O)=O)C1)CC2 Cn1ccc(=O)c(C(=O)NC2CC(CCCNC(=O)CSC3CC3)C2)c1 c1(C(=O)NC(CC)(CNC(=O)C(F)OC)CC)cccc(SC)c1[N+](=O)[O-] N1(C(c2nc(C)n(C)n2)=O)CCOC2(C1)CN(C(C1(C)CC1(F)F)=O)C2 CC(C)(C)C(CNC(C1C2CCC(C2)C1NC(C1(C)CC2CCC1O2)=O)=O)CO c1(CC)ccc(C(N2CC(NC(=O)CCNS(=O)(=O)CC)C(C)C2)=O)cc1N c1(C(=O)OC)ccc(S(=O)(=O)Nc2ccc(I)c(C(=O)OC)c2)cc1C(=O)O c1(OC)nc(C(=O)NCC(O)CCNC(c2occ(C)c2C)=O)sc1C C12(CNC(C3C(C)CCC3)=O)CCCOC1CCN(C(c1nccn1C)=O)C2 Cc1cc(C(=O)NC2CCCC2CNC(c2cc(Br)c[nH]2)=O)nc(O)n1 CCC(CC(=O)NCC1CCCCC1)NC(=O)COC(C)C N1(C(C2C(C)C2)=O)CC2CCC1C1CN(C(c3ncoc3-c3ccccc3)=O)CC21 c12cccc(n1)N2.C1(F)(C(=O)NCCCCC)CN(C(N2CC(C)C2)=O)C1 C1(F)(CNC(c2cc(SC)oc2)=O)CCN(C(=O)C(F)C(C)C)C1 CCCCC(O)C(=O)NCC1CCN(C(=O)C(c2ccccn2)C)CC1O c1(C(N2C3C(C(N4CC(C(N)=O)OCC4)=O)C(C3)C2)=O)ccc(Cl)c(O)c1 c1(CC)cc(C2CCCC2)n(C)c1C.c12cc(n(C)n1)C(=O)NC1CN(C1)C2=O CC(C)C1=NOC(C(N2CCCC2Cn2cc(-c3cnc(C4CC4)s3)nn2)=O)C1 Cc1cc(OC(F)F)ncc1CNC(=O)CC(O)c1cn(CCC#N)nn1 C1(CNC(C(C)(C)NC(=O)NCC)=O)CN(C)CCN1C(=O)CC(C)(F)F c1(OCC(=O)NCC(N(C(Cc2cc(C)[nH]n2)=O)C)C2CC2)cc(F)cc(F)c1 Cc1ccc(C(=O)NC2CCN(Cc3cc(CO)c(C)o3)C2)c(C)c1 CC1(NC(=O)NCCCOc2ccccn2)CC(C(=O)O)CC(c2ccccc2)C1 N1(C(c2cc(COC)on2)=O)CCCC(CO)(NC(=O)CCC2CC2(C)C)C1 C(=O)(C(=O)N=c1ccn(Cc2ccccc2)[nH]1)NCc1c(F)c(N)c(F)c(F)c1 N1(C(C2N(C(c3c(CC)cccn3)=O)CCN(C)C2)=O)CCCN(C)CC1C C12(C(=O)NC3CCCCN(C(c4cccc(SC)c4)=O)C3)CC1COC21CCC1 N1(C(C(C2CC2)OC)=O)CC2(CCN(C(=O)C(C)OC3CCCCC3)C2)C1 c1(OC)ccc(OC)c(CN2CCN(C(=O)C(=O)NCCN(C)C)CC2C)c1.C(C)(=O)O c1(C(N2CC3C(NC(c4c[nH]c(=NC)s4)=O)(C3)C2)=O)cc2c(cc1OC)CCC2 C(CC(C(C)C)NC(=O)Cc1ncc(C)s1)NC(C(CC)n1ccnc1)=O CC1CC(NC(=O)CSc2ccccn2)CCN1C(=O)C1=C(Cl)CCC1 C1(O)(C(=O)OCC)CCN(C(=O)C(N)Cc2cccs2)C1 n1(SCC)ccc(C(=O)NC2(C3CCCN3C(=O)COc3ccsc3)CC2)c1C CC1(C)CN(C(C2C=CCCN2C(=O)CCCC#N)=O)CCCO1 c1(CCC)ncoc1C(=O)NCC1(NC(C2CCN2S(C)(=O)=O)=O)CCOC1 C1(O)(CNC(=O)Cc2ccc(Cl)c(F)c2)CCCN(C(c2ccc(F)cc2)=O)C1 C(=O)(C(F)(CC)C(=O)OC)NCCC1CCCN(C(c2c(CCC)[nH]cc2)=O)C1 c1(C(N2CCC(CO)CC2)C(=O)NCC=C)scc(C(=O)OC)c1Cl.C(C)(C)O c1(C(N2CCNC2=O)=O)cc2n(n1)CCO2.n1(C2(C(=O)OC)CC2)cccn1 CS(=O)(=O)c1cccnc1N1CCC(NC(c2cccn3nnnc23)=O)C(F)C1 c1(C(C)C)ccccc1C(=O)NCCCN(C(=O)COC1(C)CCCC1)CCO N1(C(C(CSC)O)=O)CCC2(CCCN(C(=O)C(c3cc(C)oc3C)C)C2)C1 c1(N2CCN(C(CC)C)CC2)ncc(S(=O)(=O)NCC2(OC)CCSC2)cc1Cl Cc1nc(C2CC2)oc1C(=O)NCC(C1CC1)N(C)C(C1COC1)=O C1(NC(CN(C(COC)=O)C)=O)CCCC(NC(=O)CCn2cncn2)CC1 C1(CNC(CCCOCCC)=O)CC(C(=O)N(C)CCN(C)C)=NO1 c1(CC(=O)NCC(CCC)NC(=O)CC=CCCCCC)nc(C)c(C)[nH]1 c1(C(N2CC3C(CNC(C4C(OC)CC4)=O)C3C2)=O)cc(F)c(Br)cc1F c1(C(=O)NC(CNC(CCOCC)=O)C2CC2)csc2c(F)cccc12 N1(C(c2cc(C)nn2C2CC2)=O)CCCCC(CNC(=O)CN2CCSCC2)C1 C(=O)(C1CCCc2nn[nH]c21)NCCNC(C1(O)CCCC(C)(C)C1)=O C1(C(=O)CNC(=O)OCCNC(=O)NCc2ccccc2)CCC2(CC2)CO1 Cc1ccc(S(=O)(=O)N2CCCC2C(=O)N(C2CC2N)CC2COC(=O)C2)cc1 S(=O)(=O)(c1cnc(NC(C)Cc2cccs2)c(Cl)c1)N(C(CCSC)C)C [N-]=[N+]=NC1CCN(C(=O)C(C2(O)CCCCC2)NC(=O)C(F)=CC2CC2)C1 c1(C(=O)NC(C2CCN(C(=O)OC(C)(C)C)C2)C(=O)O)ccc(S(=O)(=O)NC)cc1 C1(NC(c2cc(COC)no2)=O)CC12CCN(C(=O)C(O)C1CCCC1)C2 C(=O)(CCCCCC(C)(C)C)N1C(C(C)NC(C2(CCOC)CC2)=O)CCCC1 c1(C(=O)NC(C)CN(C(=O)CCS(C)(=O)=O)C)cncc2nnn(C)c12 C(=O)(CCCCCCCC)Nc1ccnc(C(=O)NCCOCCOCC)c1 c1(C(=O)NC2CCC(NC(C(COC)O)=O)C2)ccc2ncccc2c1 C1(OC)CN(C)C(C)(C(=O)NCCC2(O)CN(C(c3cc(C)ccc3F)=O)C2)C1 Cc1nnc2n1CC(C(N1CCC(NC(=O)Cc3cccnc3O)CC1C)=O)C2 n1(CC)c(O)nc2ccc(C(=O)NCC3CC(NC(=O)C(C)O)C3)cc12 c1(C(N(CCN(C(C2C(CC)C2)=O)C)C)=O)cc(-c2csc(C3CC3)n2)c[nH]1 C(=O)(C(O)C(F)(F)c1ccccc1)N(CCNC(c1nc(OC)sn1)=O)C1CC1 N1(C(CCC2(C#N)CCC2)=O)CCCCC(NC(C23CCCC2CCC3)=O)C1 C(=O)(C(C)N=c1cc[nH]cc1)NC(C)CCCCNC(c1ccnnc1)=O C1(C(=O)NCc2c(CC)onc2C)CN(C(=O)C(O)C(F)(F)F)CCN1C Cc1c(-c2cn(C3CC(C(=O)OC(C)(C)C)C3)nn2)cccc1N C1(C)(C(=O)NCCC(C)(C)NC(C(C)OCCCC)=O)CC=C(C)CC1 Cc1cccc(COCC(=O)NC2CCC(NC(=O)C(O)CCN(C)C)CC2)c1 N1(C(C(C(C)C)OC)=O)CC2(C(=O)NCCC(F)=C(F)F)CC1CO2 Cc1nc(C)c(C(N2CCCC2(C)CNC(c2c(C)noc2C)=O)=O)s1 C1(C(N2CC(C)C(NC(c3cccc(C(F)F)c3F)=O)C2)=O)CC12CCSCC2 CN(C)NC(=O)CCC(=O)N1CCC2CN(C(=O)CCCCCF)CC12 Fc1cc(F)c2c(CN3CCC(F)(c4ccccc4)C3)coc2c1 C1(NC(c2cccc3c2OCO3)=O)CC2CCC1N(C(C1SCCS1)=O)C2 CC1=C(C(=O)N(C2CCC(CNC(=O)Cc3nc(C)no3)CC2)C)SCCO1 C(=O)(C(C)C(=O)N1CCC(C(=O)Nc2cc(C(N)=O)nn2C)CC1)OC c1(C(C)=O)cn(C)nc1C(=O)NCC(C1CC1)NC(c1cc(C(C)C)no1)=O C1(C(=O)NC(c2ccnn2C)C)OCCC1CNC(=O)CCN1CCCC1=O c1(CCC)c(C(=O)NCC2(O)CN(C(=O)CCC3CC3(C)C)C2)cnn1C CCC(C)C(=O)NC(CN(C)C)C(=O)NCC(F)C1CCC1 C#Cc1ccc(C(N2CCC(CC(=O)NC3CCC4CC4CC3)CC2)=O)cc1C N(C(=NCC(C)NS(C)(=O)=O)NCC1CC1)CCS(c1ccc(C)c(F)c1)(=O)=O CC(C)C(C(=O)NCC1(CN(C)C)CC1)NC(C1CSC1)=O C1(C(C)(C)C)(NC(=O)CCc2ccccc2)CC(NC(C2C(C(=O)OC)CC2)=O)C1 N1(C(CC(C)O)=O)CCc2nc(C(N3CCC(C#N)(CO)C3)=O)cn2CC1 c1(NC(C(c2cccnc2)NC(C(COC)C)=O)=O)ccc(C)c(O)c1 CCC(CC(=O)NC1C2CC3C1C3C2C(=O)N(C1CCCC1O)C)C(C)(C)C Cc1cc(O)c(C(N2CCC(CCNC(C3CCCN(C)C3)=O)C2)=O)nn1 c1(C(=O)NCC2N(C(CNC(C)=O)=O)CCCC2C)cc(O)ccc1[N+](=O)[O-] CCCCC(CNc1ncc(I)cn1)NC(c1sncc1C)=O N1(C(CSCCCC)=O)CC(NC(c2cc(C)n(C(C)C)c2)=O)C(N=[N+]=[N-])C1 CCS(=O)(=O)CC(=O)NC1CCCN(C(=O)C(F)n2cccn2)C1C c1(-c2cn(C3CC(CNC4C(C(C)C)C4)C3)nn2)ccc(F)cc1 CCCCC(O)CCC(=O)NC1CCCN(C(C2CC3CC3C2)=O)C1C c1(C(N2C(C(C)C)C(NC(C3(O)CCOCC3)=O)CC2)=O)ccc2sccc2c1 C1(NC(CC2(C(=O)OC)CCC2)=O)CCN(C(=O)Cc2ccsc2Cl)CC1C c1(C(=O)NCC(CNC(C2C(OCC)C2)=O)F)cc(OC)c(OC)c(Cl)c1 N1(CC(N2CC(F)(CNC(CN(C3CC3)CC)=O)C2)=O)CCCCC(O)C1=O NS(=O)(=O)C1CC(C(=O)NCc2cn(Cc3cccc(F)c3)nn2)C1 C#Cc1cccc(C(=O)NC(C)(CNC(=O)C(F)=CC2CC2)C2CCC2)c1 c1(C(=O)NCCC2CCN(C(C3N(CC)C(=O)CC3)=O)CC2)ccc(=O)n(O)c1 Cc1cnn(CC(=O)NCC2(O)CC(NC(=O)CC(C)O)C2)c1 c1(OCC)cc(C)c(C(N2CCC(c3ccc(F)cc3C)CC2)=O)cc1C c1(CCC(=O)NCC(C)(C)NC(CC(C(CC)C)O)=O)ccc2cnn(C)c2c1 Cc1nc(C2C(CNC(CNC(=O)CC(c3ccccc3)C3CC3)=O)C2)n[nH]1 N1(C2C3CC(C3)CNC2=O)CCCC(CF)C1.C1(SC)CCOCC1.C1(C)CC1 c1(C(=O)NC(C)Cn2cc(CCC3CCC3)nn2)c(Br)c(C2CC2)nn1C1CC1 N1(Cc2ccc(C#N)s2)CCN(C(C2CCOCC2)=O)C2CC12 N1(C(C(C2CC2)OC)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1C c1(OCC)ccc(CCC(=O)OCCCOC(c2sccc2Br)C)cc1 C1(CNC(=O)C=Cc2ccncc2)CCCCN1C(=O)CCCc1ccncc1 N1(C(CC=CC=C)=O)CC(C(N2CCCC(C#N)C2)=O)C2(CCC2)C1 C1(C)(CC(=O)NCc2cc(C(=O)NC(c3ccccc3)CC)on2)CCOCC1 Cc1cc(N2CCN(C(C3CCCC3(F)F)=O)CC2)nc(S(C)(=O)=O)n1 C1(NC(C2(COCC)CC2)=O)CCCC1NC(=O)C(C)(C)c1cnn(C)c1 CC(C)C(O)C(C)(C)C(=O)NC1CCCC1NC(c1cc(O)cc(O)n1)=O O=C1CC(C(=O)Nc2ccnc(N3CCN(C(=O)OC(C)(C)C)CC3)c2F)=NN1 c1(C(C(=O)NCC(C2CC2)NC(=O)CCc2ccccc2)O)ccc(F)cc1F CCCC(O)CC(=O)NC12CCC(C1)N(C(c1cc(O)ccc1OC)=O)C2 c1(CC(=O)OCC)csc(CS(C)(=O)=O)n1.C12CC1C(=O)N2 CC(C)C(C(=O)NCC(C(C)C)NC(=O)CCOCC(F)(F)C(F)F)C1CCC1 C1(NC(CC(CC)C)=O)CCN(C(c2cnc(OC)c(C)c2)=O)C12CC2 c1(C(=O)NC(C2CCN(C(CC3N(C)CC=CC3)=O)C2)(C)C)ccc(N)c(N)c1 CC1(C)C(NC(=O)CSc2cccc[n+]2[O-])CCN1C(C1CC1(C)C)=O C=C(C)CN=C(NCC1CCCC(F)(F)C1)NC1CC1C1CCC1 c1(C(=O)NC2C(NC(c3ccnc(C)c3C)=O)CCCC2)ccc(S(C)(=O)=O)cn1 CC(CCC(C)(C)C)C(=O)N1CCCC(N(C)C(c2ccnn2C2CC2)=O)C1 N1(C(Cn2cc(CNC(C3N(C)CCCC3)=O)nn2)=O)CC2(CCNC(=O)O2)C1 C=CCCCC(C(=O)NC1CN(C)CC12CC2)NC(c1cocn1)=O c1(CNC(CN(C)CC)=O)cc(O)nc(CNC(=O)CSc2ccc(Cl)cc2)n1 C(=O)(C(O)CC(F)(F)F)NC1(CC=C)CN(C(c2ccc(O)c(Cl)n2)=O)C1 C1(CNC(=O)C(C)n2cccn2)(NC(CC2(C)CC2)=O)CCCCCC1 c1(C(N(CC(=O)Nc2ccc(CC)nc2)C2CC2)=O)cccc2ccnn12 C1(CNC(C2CC(SC)C2)=O)CC(O)CN1C(c1cnc(S)n1C)=O c1(C(N(C(c2ccccn2)C)CC)=O)cc(Sc2cnn(C)c2)cc(Br)c1 N1(C(c2ccc(C)cc2)=O)Cc2ccccc2C(CNC(=O)CC2CCC2)C1 N1(C(C)=O)CCC2C(CCN2C(C2CCCN(Cc3ccc4c(c3)CC4)C2)=O)C1 C(=O)(CC1=CCCC1)NC(C)C(=O)NC1CC(F)CN(C(N)=O)C1 C1(C(C)C)C(C(=O)NCCCC(C)(C)C)CCN1C(c1csc(C)n1)=O c1(-c2n(C3C(C)OCC3)nc(-c3cccnc3)n2)cc2n(c1)CCS(=O)(=O)C2 C12CCN(CC1(F)F)C2=O.NC(=O)N=c1[nH]nco1.C12CC(=O)N(C1)C1CN2C1 c1(C(=O)NCC2(C)CC(NC(=O)CCSC(F)(F)F)C2)cnc2ccccn12 c1(C(=O)OC)sc(C(N2CCC(O)(CNC(c3c(C)ncn3O)=O)C2)=O)cc1C C(=O)(CCCCc1ccccc1)NCC1(OC)CCN(C(=O)COC(C)(C)C)C1 C1(C(=O)OCC)CC(N=c2[nH]c(=NC3CN(C)C3)c3c(F)cccc3[nH]2)C1 C(=O)(C1=CCCC1)NCC(C(C)C)NC(c1cnoc1-c1cccs1)=O C1(C(=O)NCC2N(C(COCC(=C)C)=O)C3CCC2C3)CN(CP(C)(C)=O)C1 C1(C(=O)NC2CCCC(C#C)C2)CN(C(=O)C(C)CO)CC1C1CC1 Cc1cc(C(=O)NC(CNC(=O)C(F)(F)c2csc(C)c2)C2CC2)co1 N1(C(c2cc(OC)ncc2)=O)CCC2(CC2C(=O)NC2CCC(F)(CO)C2)C1 C=C1CCCN(C(=O)C(CCN(C)C)NC(=O)Cc2csc(C)n2)C1 C1(NC(C(CC=C)C)=O)CC(F)CN(C(c2ccccc2Br)=O)C1 c1(C(N2CC(CNC(c3cnc(OCC)nc3)=O)(OC)C2)=O)ccnc(Cl)c1O C=CC(C)C(=O)NC(C)(CNC(=O)C(C)(C)c1ccccn1)Cn1cccn1 c1(C(N2CCCC(CCCO)C2)C(=O)NC2CCCC2CO)cccc(Br)c1 c1(C(=O)NCC(CC)NC(=O)CC2C=CCCC2)cnnc(C)c1 c1(C(=O)NCC2CC(NC(C3(CCF)CC3)=O)C(O)C2)c(F)cc(F)cc1Cl N1(C(c2nc(CC)oc2)=O)CC(NC(=O)C(C)CC(F)F)C2CCCC12 CC1C(NC(=O)C=C(C2CC2)C2CC2)CCN1C(c1cc(N)ccn1)=O c1(OCC)ccccc1NC(=O)CC1CCCCC1C C(C(=O)NC1CCC1C(=O)NC(C)(CO)C1CCCC1)(C(C)(C)C)OC CCC(CC(F)(F)F)NC(c1cn(CCNC(c2ccc([N+](=O)[O-])o2)=O)nn1)=O CCC(CC(=O)NCC1(NC(c2ccnc(O)c2)=O)CCOC1)C1CC1 C(=O)(C1=CCCC1(C)C)NCC(CC)(CC)NC(C1CCN(C)C1=O)=O N1(C(C(COC)C)=O)CC2CC2(NC(c2ccc(-c3nccn3C)cc2)=O)C1 C1(C(C)(C)CNC(c2cnsc2)=O)CCCCN1C(C1CC(=O)N(O)C1)=O C=CCC(C)(C)CCNC(C1(NC(C2CC(=O)C2(C)C)=O)CCSC1)=O C#CCN=S(C)(=O)NCCCC(F)(F)Br.c1ccccc1 C1(NC(=O)CNC(c2cn[nH]c2)=O)CCOCC1NC(C1CC(F)(CO)C1)=O C1(C(N2CC(CNC(=O)C(C3CC3)C3CC3)C2)=O)CCCCS1(=O)=O c1(CC)c(C(=O)NCC(c2ccccc2)Nc2nccc(SC)n2)cnn1C Cc1cc(Cl)cc(C(N2CC(C(N3CCC(C)C3)=O)CC(F)C2)=O)c1O c1(C(=O)NCC2(C(=O)NC3CC4(CCC4)C3O)CCC2)cccc2cncn12 C(=O)(CCCCC(N)=O)NCC(COc1ccnc(Sc2ccccc2)n1)OC C1(CNC(c2c(C)cno2)=O)CCC2CN(C(=O)C=CC(=O)N(C)C)CC12 C1(S(C)(=O)=O)(C(=O)NCC(C)(C2CC2)NC(COCCOCC#C)=O)CC1 C1(C(=O)NCC(CCC(C)C)C)CC(O)CN1C(=O)C(c1ccnn1C)C C1(O)(C(=O)NC(C2CCN(C(c3cc(=N)[nH]n3C)=O)C2)C)CCCCCC1 c1(C(N2CC3(C(NC(CCC)=O)CCS3)C2)=O)ncnc2c1cnn2C C1(NC(CC(CC)CC)=O)CCC2(CC1)CC(NC(=O)C(CO)OC)C2 CC1CC(O)CCN(C(=O)CCCCN(C)C(C2(C)COC2)=O)C1 CC(N=c1nc[nH]s1)C(C1CCCC1)NC(=O)CCc1nccn1C C1(NC(C(CC)c2ccccc2)=O)CC2(CCCN(c3ccnc(Br)n3)C2)C1 c1(C(=O)NC(C)CN(C(=O)COC2(C)CCCC2)C)cc(Cl)nnc1O.OCC c1(NCCC(=O)NC(C)C)cc(=NCCc2cnccc2C)[nH]cn1 CCCC(CC1CCC1)C(=O)N1CCCCC(NC(c2c(C)ncn2OC)=O)C1 c1(C(=O)NC(CCOCC)C(=O)NCC2(CO)CC2(C)C)ccc(F)cc1F c1(C(C(=O)NCC)N(C)Cc2ccc(NC(=O)N(C)C)cc2)cc(C)nc(C)n1 c1(C(=O)NCCN(C(C2(C)C(C)CCC2)=O)C)ccc2c(c1)C(=O)N(C)C2 N1(C(C(C)OC)=O)CCN(C(c2ncccc2O)=O)CC1c1ccccc1F C1(C(=O)NCC2(NC(c3cnc(COC)s3)=O)CCC2)C(C)(C)OC1(C)C C1(F)(NC(c2ccc(OC3CCC3)cc2)=O)CCOCC1 c1(C(=O)NCCN(C(c2c(C)cnn2C)=O)C2CC2)cc2cccnc2cc1F N1(C(c2n(CC#C)ccc2)=O)CCC2CC1CN(C(=O)CNC(N)=O)C2 c1(C(N2CC(NC(C(C)CN(C)C)=O)C(C)C2)=O)cc2c(O)ccc(F)c2[nH]1 C#CCC(CC(=O)NCCC(CO)C(C)C)NC(=O)C=CC=CCC c1(C(=O)NC(C(C(C)C)C)CNC(=O)C=CCO)cc([N+](=O)[O-])cnc1O c1(C(=O)NCCCCNC(C2C(C)(Br)C2)=O)ccc(OCC(F)F)cc1 C1(NC(C(CC#C)O)=O)CCN(C(c2nc(CC)ncc2Cl)=O)CC1F c1(C(=O)NC(CSC)(C)C)ccc(CNC(=O)C=Cc2ccc[nH]2)o1 C1(C)(CNC(C(CC2CCC2)OC)=O)CC(F)(F)CN1C(=O)C(C)OC c1(C(=O)NCC(CC=C)NC(=O)C(F)C(F)(F)F)oc2ccccc2c1Cl N1(Cc2c(C)c(Cl)ncc2)CC2OCCN(C(c3ccccc3Cl)=O)C2C1 Cc1cn2c(n1)CCC(C(=O)NCCNC(c1ccc(C)c(F)c1F)=O)C2 N1(C(Cn2nc(C)c(Cl)c2)=O)CCN(C(=O)Cc2cnccn2)CC(C)C1 CCCC(C)CCN=c1[nH]c2c(c(=NCC(C3CCOC3)OC)[nH]1)CSC2 C(=O)(CS(=O)(=O)C1CCCC1)N1CCC(C2CC2)(NC(C(COC)C)=O)C1 C1(NC(Cc2cc(C)on2)=O)COCCC1NC(C1(Cl)CC12CCC2)=O C1(NC(C(C)N2CCC2)=O)CC2CC1N(C(=O)Cc1ccnc(Cl)c1F)C2 Cc1c(Br)ccnc1N1CCN(C(=O)C(N2CCCC(O)C2C)=O)CC1 C1(CC#C)(C(N2CCC(C(C)NC(c3cn(CC=C)nn3)=O)C2)=O)CCCC1 N1(C(C(CN(CC)CC)F)=O)CCC2(CCC(NC(C3CN(C)C3)=O)C2)C1 c1(C(=O)NC(CC(C)NC(CCCC)=O)C)c(OCCCOC)cccc1Cl c1(CNC(C(C)NC=O)=O)cc(C(=O)NC(c2ccccn2)C)cs1 Cc1cc(CNC(=O)C(C2CCOC2)C2CC2)ccc1O.C12(CCCO1)C(=O)N2 C(CCS(=O)(=O)c1ccccc1)NC(CC1(N)CCSC1)=O C(=O)(C1=CC2CCC1C2)N1CCN(C(c2scc(C#N)c2)=O)CC1CC(F)F c1(OC)cccc(CCC(N2CCC(CNC(=O)COC3CC(F)(F)C3)C2)=O)n1 N1(C(C=COCC)=O)CCC2(CCCC2C(=O)Nc2ccc(C3CC3)cc2)C1 c1(C(=O)NCC2N(C(C(CC#C)C)=O)CCCCC2)nc2c(s1)CN(C)CC2 C12(NC(=O)CC3CC(F)(F)C3)CCN(C(c3ccc(O)c(F)c3F)=O)CCC1C2 C(CC(=O)NC1COC(C(C)C)C1)(C(F)(F)F)NC(c1c(OC)scc1)=O c1(-c2nc(N(C(c3cccc(C(=O)OC)c3)=O)CCO)on2)c(F)cccc1F N1(C(C(c2ccccc2F)(C)C)=O)CC2(CCC2NC(C2C=CCC2)=O)C1 c1(NC(=O)NCC2N(C(CCCSCC)=O)CCC2)ccc(Cl)c(S(C)(=O)=O)c1 C1(C#N)(C(=O)NCC=CC(=O)NC(COC)CO)CC2CC2C1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CCCC(F)(F)F)CC12CCC2 C1(CNC(CC2C(C)C2(F)F)=O)CN(C(C2CC(=C3CC3)C2)=O)CCCO1 c1(NC(COC(CNC(C(n2c(C)ccn2)C)=O)(C)C)=O)cnccc1C1CC1 N1(C(CCc2ccc(C)o2)=O)CCOCC(CNC(=O)CN2CC(C)(C)C2)C1 CC1CCN1CC(=O)N(CCO)CCOCCO CCCCC(F)C(=O)NCC1CCC(NC(C2CCCN(C)C2)=O)CC1 C(=O)(NN1CCCC(C(=O)O)C1)C1(N=[N+]=[N-])CCCN(CC)C1 N1(C(CC(CC)(F)F)=O)CCCCC2(CCN(C(C3CCC4(CCC4)O3)=O)C2)C1 N1(C(CC(CC)OC)=O)CCCC(C2CCN(C(=O)CCc3cnc(C)o3)C2)C1 c1(CCC(=O)N(C(CCNC(CCOCCOCC)=O)C)C)cnc(C)s1 c1(C(CNC(=O)NC2(Cc3cccs3)CCC2)O)noc2ccccc12 C(=O)(C(C)CC(=O)NCC1CCCN1C(C1CN(CC(F)(F)F)C1)=O)OC N1(C(C(C)C#N)=O)CC2(CCC(CNC(=O)C=Cc3ncc[nH]3)O2)C1 N1(C(C2N(C(C(C)S(C)(=O)=O)=O)CCSC2)=O)CC2(C)CCC2(C)C1 N1(c2ncc(C(=O)OCC)s2)CC2CCCN(C(c3cnn[nH]3)=O)C2C1 c1(C(N(CCCCNC(=O)Cc2ccn(C)n2)C)=O)ccccc1C1(C)CC1 Cc1nn(C)cc1CCC(=O)NC1CN(C(C2CC2C(F)F)=O)C1 C(CC(=O)NC(C)CNC(c1csc(C(C)OC)n1)=O)(C1=CCCC1)OCC C(=O)(C(C)(C)C1=CCSCC1)NCC1CCC(NC(C2(C)COC2)=O)C1 N12CC(CC(C)C1)C2=O.N1(CC=O)CC(=O)N(C)C1=O.N1(CC)CCN(CC)CC1 Cc1ccc(I)cc1Cn1cc(C2(Cc3ccccc3)CCCO2)nn1 C=CC1CN(C(=O)C(CCC)NC(N)=O)CC1NC(c1ccc(N)cc1CC)=O CC(CNC(c1cn(C)nn1)=O)CC(=O)NC1CC12CCCC2 C1(CNC(C(C=C)O)=O)C2CCCC1N(C(C1CCC(C)O1)=O)C2 Cn1ccnc(NC(c2cccc(C(c3ccccc3)=O)c2)=O)c1=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC1N2C(=O)CC(C)c1ccco1 N1(C(c2c(C(C)C)nn(C)c2)=O)CCC2C1CCCN2C(=O)CCC1(C)CC1 c1(NC(C(CC)NCCO)=O)ccc2nc3n(c(=O)c2c1)CCCC3 C12(O)CCCN(C1)C2.Cc1onc(C(=O)CCNCc2cncc(C(C)(C)C)c2)c1C CC1Cc2sc(C(N3CC(NC(c4cccc(F)c4Cl)=O)C3)=O)cc2C(C)C1 N1(C(c2cc(OC)nn2C)=O)CCN(C(C2CCC(=O)N2)=O)CC1c1ncc[nH]1 CC(C)(C(=O)NCCCC1CCOCC1)NC(=O)CC1COCCO1 C1(NC(CCC(=C)Br)=O)CCC2(CC1)CN(C(c1cc(C)[nH]n1)=O)CCO2 c1(C(N(C(C)CCNC(c2c[nH][nH]c2=N)=O)C)=O)ccc2c(O)n[nH]c2c1 c1(CC)ccc(C)c(C(=O)NC2(CCCNC(=O)C(O)C(C)C)CC2)c1 Cc1cc(C)c2cc(C(N3CCCC3CNC(=O)C3=CCC(C)CC3)=O)[nH]c2c1 CCCC(CC(=O)N=c1cc(CC2CCCCC2)[nH][nH]1)N(C)C C(=O)(CN=S(C)(C)=O)NC1C(NC(C(c2ccc(OC)cc2)CC)=O)CCCC1 C1(CNC(C=CC=CC)=O)CCCC(CNC(c2cc(CC)ncn2)=O)C1 Cn1cc(CCC(=O)NCCC2(C(=O)NC3(C(O)CO)CC3)CCCC2)nn1 C(=O)(C1=NOC2(CCOC2)C1)N1C(CNC(c2ccn(CCF)n2)=O)COCC1 CCC(O)C(C)C(=O)NCC1CC(NC(c2cn(C)cc(Br)c2=O)=O)C1 N(C1COc2c(Br)cccc21)C(N1CCc2cc(Cl)ccc21)=O C(N=c1[nH]c(=NCC2CCCCS2)c2ccccc2[nH]1)C1C(C(C)C)OCCC1 C1(O)(CCNC(c2csnn2)=O)CCN(C(c2ccc(O)c(F)c2)=O)CC1 c1(CC(=O)NCCC)cn2c(C)ccc(-c3cccc4c3CCC4)c2n1 c1(OCC)cc(C(N2CCC(NC(C3CC3C)=O)C2)=O)ccc1OCC c1(N(CC(CCC)C)C)nc(=NC(C)c2nnc(COC)s2)[nH]c2c1CCC2 C=CC(CCC)CC(=O)N1CC(OC)CC1CNC(c1cnn2ccn(C)c12)=O C1(c2n(CC)nnn2)(NCCSc2ccc(CN(C)C)cc2)CCC1C1CCC1 N1(C(c2ccc(NC)cn2)=O)CC2(CCC(CNC(=O)CC=C(C)C)O2)C1 c1(C(C(N2CCC(N(CCC)C(C)=O)CC2)=O)=O)ccc(C(=O)NC2CC2)cc1 c1(C(=O)NCC2CC(NC(CSC(C)C)=O)C2)cc2c(OC(F)F)cccc2[nH]1 Cc1csc(C=CC(=O)NCC23CC2CN(C(c2nc(C)oc2C)=O)C3)n1 C1(CNC(C(F)OC)=O)CCN(C(c2ccc(C)nc2O)=O)C12CC2 N1(C(C2CN(C)C2)=O)CC2(CO)CC1(C(N1CCC=C(F)C1)=O)C2 c1(C(N(C2CC2)CC2C3CN(C(=O)CC(F)(F)F)CC32)=O)cc2sccc2[nH]1 C#Cc1cc(C(N2CCC(CNC(C3(c4ccn(C)n4)CC3)=O)C2)=O)cc(Cl)c1 N(C1CCN(C)c2ccccc21)C(c1ccccc1CO)C C1(CCC)CN(C(=O)CCCN(C)C)CC1C(=O)N(CCN1CCCC(O)C1)CC N1(C(C(CCC)OCC)=O)CCC2(CCC2)C(NC(c2oc(C)nc2C)=O)C1 C1(C(C)C)CN(C(C2(F)CCN(C(=O)CC3(C)CCOCC3)CC2)=O)CCCO1 c1(OC)ncc(NC(C2(C)CCCN2C(=O)CN2CCOC2=O)=O)cc1Br c1(OCC(=O)NCCCCNC(=O)CC2CCC3CC23)cccc(F)c1F C1(C(N(C(CCNC(C2ON=C(CC)C2)=O)C)C)=O)CC2CCC1CC2 c1(OCC(N)=O)ccc(CC(=O)NC2CC(NC(=O)C(F)(F)SC3CC3)C2)cc1 C(=O)(C(C)CC(C)(C)C)N(CC(C)N(C(CCNC(=O)OC)=O)C)C c1(CCNC(C2CC2Cl)=O)c[nH]c2ccc([N+](=O)[O-])cc12 c1(C(=O)NCC2(C)N(C(C3=C(C)CCCC3)=O)CCC2)cccc(O)c1[N+](=O)[O-] c1(C(N(CCC)CCN(C(=O)CC2CC2C)CC)=O)ccc(OCC(F)F)nn1 N1(C(c2ccc(CC)nc2)=O)CCC(O)C(C(=O)Nc2ncc(O)cc2Cl)C1 c1(C(N2CC(OC)(CNC(c3ncn(C(C)C)n3)=O)C2)=O)cc(F)cc(C)c1N N1(C(C(C)N2CCC2)=O)CCOCC(F)(CNC(=O)CCc2cn[nH]c2)C1 c1(OC)ccc2[nH]c(=NCCc3ccccc3Br)[nH]c(=NCc3cnn[nH]3)c2c1 CCC(CC(=O)N1CCCC(CC)(NC(=O)CCSc2ccccc2)C1)C(F)F Cc1cnc(CN2C(C(N3CC4(CCC4)C3)=O)CC3CC23)c(F)c1 c1(C(N2CCC(C3N(C(C(F)OC)=O)CCC3)C2)=O)nc(Cl)sc1Cl c1(C(N2C3C(NC(CC(C)CF)=O)C(CC3)C2)=O)c(C2CC2)nc2sccn12 Cc1ccc(CCCn2cc(CN(O)C(=O)NCSC3CCCC3)nn2)o1 C(=O)(C(C)(C)C(C)(F)F)NC(C1CC(NC(c2c(C)occ2)=O)C1)C C1(NC(c2c(C)[nH]nc2Cl)=O)CCN(C(=O)CSC2CC2)C(C2CC2)C1 C1(C(=O)NC(C)CCNC(=O)CC2CC2(Cl)Cl)CCOC2(CCCCC2)C1 C1(CC=C)(C(N2CCC(N3C(=O)CCC3=O)CC2)=O)CNCCO1 Cc1ncc2cc(C(=O)NC(C3CCCN3C(=O)CC(C)CC(C)C)C)ccn12 CCCC(CC)C(c1nnnn1CC(F)F)NCc1cnccc1C CC(C)(CNC(=O)C=CCNC(c1n[nH]cc1Cl)=O)C1=CCCC1 C1(NC(=O)Cc2cc(F)ccc2F)CC12CCN(C(=O)Cc1nnc(O)s1)CC2 CC1(C)CC(CC(=O)NC2CC(CNC(c3cc(Cl)c[nH]3)=O)CC2O)CCO1 C(=O)(CCCCC(F)F)NC(C1CCOC1)CNC(=O)Cc1nnc(O)s1 c1(C(N2CC(O)CC(NC(C(C)(C)N3CCCC3)=O)C2)=O)ccc(F)c(Cl)c1F c1(CCCC(=O)NCC(CNC(=O)C(C)SC)OC)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)CO)cccc2occc12 C(=O)(CN=c1cc[nH]cc1)N1C(NC(C(C)Oc2ccccc2Cl)=O)CC(O)C1 C(CCC(=O)N=c1ccn(Cc2ccccc2)[nH]1)C1C(C)CCC1 CC(C(F)C(=O)NCCC1CN(C(c2sccc2C2CC2)=O)C1)C(F)(F)F c1(CC(=O)NCCC(=O)NC2CN(CC)CC2C)cccn2cncc12 C1(C(N2C(C)(CCC)CC2)=O)CC(C)CCN1C(c1cc(O)nn1C)=O C1(CN(C(=O)C(=O)NCc2ccc(Br)cc2F)CC)CC12CCOCC2 c1(C(=O)OC)cc(C)c(C(N2CC(CNC(c3cnn(C(C)(C)C)c3)=O)C2)=O)o1 c1(C(=O)NC(CCOC)CNC(=O)C(c2ccccc2)F)cccc(=O)n1C c1(OC)ccc(C(=O)NCC2CCC(NC(=O)CN3CCCCC3)C2)c(F)c1Cl CC(=O)CCCC(=O)NC(C(=O)NCc1cc(=O)cc[nH]1)C(C)C c1(C(=O)NCC(CC)NC(=O)CC2CNC(=O)O2)ccc(C)c(C)c1F N1(C(c2c(OC)cccn2)=O)C2COCC1CC(NC(=O)COCCCF)C2 c1(C(C)NCc2cn(C3COC(C)(C)C3)nn2)cnn(-c2ccccc2)c1C1CC1 CC(CS(=O)(=O)Nc1ccc(N2CC(O)C2)cc1)C(F)F c1(CNC2CC(CC(=O)NCc3c(C)ncs3)C2)cc([N+](=O)[O-])c(Cl)cc1F N#Cc1c(Cl)nc[nH]c1=NCC(CNC(=O)C=Cc1ccccn1)C(F)(F)F N1(C(CC2C(C)C2)=O)CC=C(CNC(=O)CCCc2ccc(F)cc2)CC1 C1(NC(C(C)O)=O)CN(C(c2ccc([N+](=O)[O-])cc2)=O)C2CCCC12 c1(C(=O)NCC2CCCCN(C(CCC(C)(C)F)=O)C2)cc2n(n1)CC(F)C2 c1(C(=O)NCC2CCCC2)c(-c2ccc(F)cc2Cl)ccc2c1OCO2 C1(NC(c2n(C)ccn2)=O)CN(C(=O)C(C)(C)C(N)=O)CC12CCC2 C(=O)(C1=NOC(CNC(C2CNC(=O)N2)=O)C1)N1C(C)(CCC(=O)NC)CCC1 C(C)(CC(=O)NCC1CSCCO1)NC(CC1(NC(C)=O)CC1)=O CCC(CCCC(=O)NCc1noc(C(N)=O)n1)NC(C1CCOC(C)(C)C1)=O C12(NC(c3c(C)nc(CC)s3)=O)CC(CNC(=O)C=C(C)C(C)(C)C)(C1)OC2C CC1(C)CCCC(C(N2CCC(C(F)F)C2)=O)C1 N1(C(c2sccc2F)=O)CCN(C2CCN(C(c3[nH]nnc3C3CC3)=O)C2)CC1 C1(C(=O)NCC(CC)NC(=O)C=C2CCC(C)C2)(OCC)CCCCCC1 CC(C)(CCCNC(C1CC(C)(C)C1)=O)NC(C1CC1C(F)(F)F)=O c1(OC)ccc(Cl)c(C(=O)NCCC2CCN(C(c3cn(C4CC4)cn3)=O)C2)c1 C1(C(N2CCN(C(CCOc3ccc(OC)cc3)=O)CC2)=O)CCC=CCCC1 CC1C(NC(C2CC3CC3CC2C)=O)CCCN1c1nccc(CC#N)n1 C12(CNC(C3(C)CCCOC3)=O)CCC(CC1)N(C(C1CCN1S(C)(=O)=O)=O)C2 Cc1ccc(OCC(=O)NC(CNC(c2ccc(=O)n(C)c2)=O)C2CC2)c(Cl)c1 N1(C(C2C(C)(C(F)F)C2)=O)CC(CNC(=O)Cc2ccsc2)C2(CCOCC2)C1 N1(C(C(C)(C)SC)=O)CCCCC1c1cn(-c2c(C)cnn2CCO)nn1 n1(CC)nc(C)c(C(=O)N(CCNC(c2cncc(C(C)(C)C)c2)=O)CC)c1C N1(C(CCCCCCC)=O)CC2COCC(C1)C2NC(c1coc(CC)n1)=O C(=O)(N=c1ccn(C(C)C)[nH]1)C1(CC)CCN(C(=O)CC2(C)OCCO2)CC1 CCCC(CCC)=CC(N1CC(F)(CC(=O)NCC2CC(=C3CCC3)C2)C1)=O c1(C(=O)NC(CC)(CC)CC)ccc(C(F)(F)F)nc1C N1(Cc2nnc(COC)s2)CCC(c2ccccc2)CC1C C=CC(C)(C)CCCNC(c1cc(CNC(=O)C2=CCOCC2)no1)=O N1(C(CCN(C)C(c2csc(O)n2)=O)=O)CCC(CN=[N+]=[N-])CC1 C(=O)(C1=CCCN(C(=O)Cc2cncnc2O)C1)N(C1CC2CCC1C2)C CC1(NC(c2ccc(C(F)F)cn2)=O)CCN(C(=O)C=CC(N)=O)C1 C(=O)(C(C#N)C(C)(C)C)N1C(C(=O)Nc2cccc(C)c2F)C(C)(C)CC1 c1(CC)cnc(Cl)[nH]c1=NC1CCCN(C(=O)Cn2nc(C)cc2C)CC1 C(=O)(C(C)(CO)NC(=O)Cc1ccoc1)N(C(CC)CC)C C1(NC(c2c(CC)oc(C)n2)=O)CC12CCC(NC(=O)CCNC(=O)OC)CC2 c1(CC)ncccc1C(=O)NC(CCF)C(=O)NCc1ncsn1 c1(NC(C2CCN(C(c3c(C)oc(Cl)n3)=O)C2C)=O)ccc(O)c(Cl)c1 CC1CN(C(C2CCC(CNC(=O)Cn3ncn(C)c3=O)CC2)=O)CCCO1 Cn1ncnc1CCCNC(=O)C=CCNC(=O)CC1(CO)CCC1.C(C)(C)(C)O C(CC(=O)NNC(=O)c1ccco1)(C(=O)OC(C)(C)C)SC O=C(N=c1ccc(Cl)n[nH]1)C1=NOC2(CCN(C(c3csnn3)=O)C2)C1 c1(C(N2CC(C)C(CNC(c3ccnc(CO)c3)=O)C2)=O)ccn2ccnc2n1 c1(CN2CCCC(C(=O)NC3CC(F)C3)CC2)c(O)cc(O)cc1O c1(C(N2CCC(N(C(C)=O)C(C3CCCO3)C)CC2)=O)ccc(O)c(CO)c1.CCO c1(C(=O)NC2CCC(CNC(c3c(NC)nccc3)=O)C2)ccnc(O)c1F C1(C(N2CC(O)(C(C(=O)NCc3scc(C)n3)F)C2)=O)CCC(=O)NC1 Cc1ccc(F)cc1C(N1CC(C)(C(=O)Nc2c(Cl)n[nH]c2C)C1)=O c1(C(=O)NCC2C(NC(C3ON=C(C(C)C)C3)=O)COC2)ccn2ncnc2c1 c1(Cc2nc(-c3ccc(OC)nc3)nn2CC2CCCO2)ccccc1S(C)=O C12(C(=O)NC3CCN(C(C4(CC=C)CCCC4)=O)CC3)CCC(F)(CC1)CC2 c1(C(=O)NC2CCCN(C(C3(C)CCN(C)C3=O)=O)C2)ccc2oc(S)nc2c1 C(C(COC)CC(=O)N1CCN(C(C2C=CCC2)=O)CC1CCO)OC CCCCC(CC(=O)N1CCCCC1CO)NC(=O)C(C)=CC1CC1 N1(C(C=CC(CC)C)=O)CC(CNC(=O)CCCC2CCC2)(OC)C1 c1(C(=O)NC(C)(C)CNC(C2CC3CCCC3C2)=O)cncc([N+](=O)[O-])c1 CC1CN(c2nc(N3CC4CCC(C3)N4C)c3ncsc3n2)CCC1(F)F c1(CN2CCN(C(C(C)OCCCC)=O)C3C2C3)cc2c(OC)cccc2s1 N1(C(C(C)O)=O)CCCC(NC(c2nnc(S)n2C)=O)C1C CCCC(C(=O)NCC(CC)(CC)OC)NC(c1ccccc1OC)=O C(N=c1cc(NCC2(COCCO)CCOC2)nc(C)[nH]1)c1ccc(SC)o1 Cc1cc(N)cnc1C(=O)NCCCCC(C)NC(C1(CO)CCCCO1)=O C(=O)(CC1OCCc2ccsc21)NC(C)CNC(=O)CSCc1ccnn1C N1(C(C2C(=C)C2)=O)CC(NC(=O)CC2CCS(=O)(=O)C2)CC1C c1(C(C)C)cc(CC(=O)NCC(C)(F)CNC(C2(CF)CC(=O)C2)=O)on1 C(=O)(CC(CN(C)C)C(F)F)NCC(C)(C1CCC1)NC(c1c(C)cccn1)=O C1(CCC=C)(C(=O)OC(C)(C)C)CN(C=O)C1.C(CCSC)(c1nn[nH]n1)NCC Cc1nc(NC2CCCN(C(=O)C(O)Cc3ccc(O)cc3)C2)c2sccc2n1 c1(C(=O)NCC2N(C(CC(=O)OC)=O)CCOC2)c(Cl)c([N+](=O)[O-])nn1C C1(CC(=O)NCC2(OC)CCN(C(C34CCC3CC4)=O)C2)CCCCC1(C)C C(CO)(C(C)NC(=O)C(CO)NC(=O)C(F)(F)F)NC(C=CC(=O)N(C)C)=O c1(C(=O)NCC2N(C(c3cc(CC)oc3C)=O)CCC2)cc2nc[nH]c2cc1F N1(C(c2c(C)nc(C)o2)=O)CC(CNC(=O)C(O)CN(C)C)CC12CCC2 CCC(C)CC(=O)NCCCCSC.c12nn(cc1Br)c(=O)[nH]2 c1(CCNC(c2cc(OC)c(C#N)cc2)=O)cnc2ccccc2c1 CC1CCC(CNC(c2cccc(O)c2F)=O)CN1C(c1cncs1)=O c1(C(N2CCC(N(C(=O)Cc3ccc(F)cc3)C)C2)=O)coc2c1CSC2 C1(NC(c2c(CC)non2)=O)CCC2(CC1)CC2NC(c1ccnc(OC)c1)=O C(CC(N)=O)(C(=O)N(C1CCCC(O)C1)C)NC(c1c(CC)n(C)cc1)=O N1(C(c2c(COC)ncs2)=O)CCCC2CN(C(=O)C(C)(O)C(C)C)CCC12 CC(C)C(F)(CN)C(=O)N(c1ccoc1)C1CC1 Cc1cc(F)ncc1CN1CCC(O)C(C(=O)NC(C)CF)C1 C#Cc1cnn(C)c1C(N1CCC(CC(=O)NCCc2ccc(F)cc2)CC1)=O c1(C(=O)NCCN(C(=O)CC2CCOC(C(C)C)C2)CC)ccc2c(c1)CCC2 O=C1Cc2cc(S(=O)(=O)NC3CC3c3cc(Cl)cc(Cl)c3)ccc2N1 c1(C(=O)NC2CC(CNC(=O)C=CC3CCCC3)C2)cc(CO)ccc1Cl C1(C(C)NC(C2(C3CCCO3)CCCC2)=O)CCCN1C(=O)CC1(N(C)C)CC1 c1(C(N(CCN(C(=O)C(C)SC(F)(F)F)C(C)C)C)=O)occ2c1CCCC2 N1(C(COCCCC)=O)C2CCC1CN(C(c1ccno1)=O)CC2 C1(C(=O)NCc2ccc(C(=O)NC3CCN(CC)C3)o2)CC(F)C(=O)N1 c1(C(N2CCN(C(C=Cc3c(C)nsc3)=O)C(CF)C2)=O)cc2c([nH]1)CCCC2 c1(C(N2CCN(C(c3nccc(CC)c3)=O)C3C2C3)=O)ccc2nccnc2c1 CC(CC1CC1)C(=O)N1CC(C(N)=O)(CNC(=O)COc2ccon2)C1 CC1CN(C(=O)C(C)(C2CCC2)NC(=O)C=C2CCOCC2)CCC1O C1(C(N(CC(CC)C)CC)=O)CN(C(c2cc(C)oc2C)=O)CC1(F)F C12CC3(CCN(CC3)C(=O)C1C(=O)OC(C)(C)C)C2.Cc1snnc1CO CC1(C)CCCCC1C(=O)NCC(CO)NC(c1cc(O)cc(O)n1)=O C12(C(N3CCCC(C)C3CO)=O)CCC(CC1)N(C(=O)C(O)C1CCCC1)C2 N1(C(C2OCCN(C(C)C)C2)=O)CC(CNC(=O)CCC(F)(F)F)OC(C)(C)C1 C123CC(CO)(CN1C2=O)C3.CCC1CC(=O)N1C1CC1.C1(C(=O)OC)CCCC1O Cc1ccc(C(=O)NC2CC2CNC(c2ccc(C#N)s2)=O)cc1[N+](=O)[O-] CC1(C)CC(S(=O)(=O)N(CC2=CC=C(OCCO)C=CC=C2)CC)CO1 C1(Nc2cc(C)ncn2)CN(C(C2CCN2C(C)(C)C)=O)CC1(C)C Cc1ncnc(C)c1CC(=O)NC(C)C(C)NC(=O)COc1ccc(O)cc1 c1(C(C(=O)NCC2CCCO2)N(C2CC2)CC)cccc(OC)c1 C#Cc1cnc(N2CCCC2CNC(C2CC2C2CC2C)=O)nc1 N1(C(c2cnco2)=O)CC2CN(C(c3c(O)cccc3Cl)=O)CC2C1 Cc1ncnc(C)c1CC(=O)NCC(CO)NC(=O)C(c1cccnc1)O C1(NC(CSCc2cccc(C)c2)=O)COCCN(C(=O)CC#N)C1 c1(OC(C2CCC(=O)O2)=O)ccc2nc(C(=O)OC)[nH]c2c1 N1(C(C2(CF)CCN(C(CCCOC)=O)C2)=O)CC2(C1)OC(=O)NC2C C1(C(=O)NC2CC3(CC(NC(c4n(CC)ncn4)=O)C3)C2)CCC2(C1)CC2(F)F C=CCC(CCCCC)C(=O)NC12CCC(CNC(=O)C(=O)NOC)(C1)OC2 C1(C(N2C(C)CC(N(C(C)=O)Cc3ccccc3)C2)=O)CCc2nnc(O)n2C1 c1(C(C)(C)C)ccc(C#N)c(NC2CN(C(C3CCCC(F)C3)=O)C2)n1 Cc1ccccc1-n1cc(CNC(=O)NCCC(c2ncc[nH]2)O)nn1 C12(Cc3nsc(-c4ccccc4)n3)CCN(CC1)C2=O.N1(CN)C2CCC1CC2 C(=O)(CCCC(N)=O)NC1CCN(CCNC(c2ncc(C)nc2)=O)CC1 c1(C(N(CCCNC(=O)CC2CC(N(C)C)C2)C)=O)cnn2c1OCC2 C12(C(=O)NCCOC3CCN(C(c4c(C)nsc4)=O)C3)CC1Cc1c[nH]nc12 Cc1nc2cc(C(N3CC4C(CNC(C5CC5F)=O)C4C3)=O)cnc2[nH]1 Cc1cc(C)c(C(=O)NC2COCC2NC(C2CCC=CCCC2)=O)c(C)n1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC(C)CN(C(=O)CC1CC1C1CC1)C N1(C(Cc2cnc(C)s2)=O)CC2CC1CN2C(c1snc(C)c1N)=O N1(CC)C(=O)CCC1CC(N1CC(CNC(=O)C=CC(C)(C)C)C(O)C1)=O N1(C(CC)=O)CC(NC(c2nccn2C2CC2)=O)C(SC)C1 C(C(C)(O)CC(=O)N1CC(CCO)(NC(c2cc(C)nc(O)c2)=O)C1)OC C1(C(=O)N)CCC(=O)CC1C.C(=O)(C(C)=CCNC(=O)CC1(CO)CC1)OC C1(NC(C(C(CNC(C2(CC)CCCCC2)=O)C)F)=O)CC2C(O)C(O)CC12 C1(C(=O)NC2(C3N(C(CCC=C=C)=O)CCC3)CC2)CCCC(F)(F)C1 C1(CNC(c2ccc(OCC#C)cc2C)=O)CCOCC12CCC2 C1(CC)(CC)CC(C(=O)NC2CCCC2C(=O)NCC2CCC(C(N)=O)O2)C1 N1(C(=O)CSCc2cccnc2)CC2CCN(C(C3CCCC3C3CC3)=O)C2C1 c1(C(=O)NCC(C)NC(C(c2ccc(C)cc2)C(C)C)=O)nc2ncccn2n1 c1(C(N2CC3C(C2)N3C(C2(c3cccs3)CC2)=O)=O)ccc(Br)c2ncccc12 c1(C(=O)NCCCCCN(C(CCN(CCC)C)=O)C)sc2ncccc2c1N c1(SC2(CNC(=O)NCCc3cc(C)no3)CC2)cncc(C#N)c1 c1(CC)ccc(Oc2nc(SC)co2)cc1.C12CN(C1)C(=O)C(=O)NC(=O)N2 Cc1cccc(Cl)c1CC(CCC(C(=O)O)N)=O N1(C(C(C(CC)O)C)=O)CCOC2(CCN(C(c3ccnc(C(F)F)c3)=O)C2)C1 C1(F)(CNC(=O)OC(C)(C)C)CCC(CNc2nc(Cl)c(C(=O)O)s2)CC1 C=CC(C)(O)C(=O)NCC(O)CC(=O)NCCC(C)C(=O)OC N1(C(CCC(=C)Cl)=O)C2CCC1CC(N(C)C(c1ccc(Cl)c([N+](=O)[O-])c1)=O)C2 CCC(CNC(c1cc(OC)ccn1)=O)N=c1cc(C2CC2)nc(Cl)[nH]1 c1(C(N2C(CNC(C3(CC#C)CC3)=O)CCCC2)=O)n[nH]c2cc(OC)ccc12 c1(N(CC(C)C)C)ccc(C(=O)NC2CCCC2NC(=O)Cn2cncn2)cn1 C1(CNC(CCN(S(CC)(=O)=O)C)=O)CCN(C(=O)CC2(O)CCCOC2)CC1 c1(CN(C)Cc2cncc(OC)c2)cc([N+](=O)[O-])ccc1F C(=O)(CC(C)C(C)(C)NC(=O)C(COC)OC)N(CC(CC)OC)C C(=O)(C(C(C)C)N(C(=O)C(CNC(=O)C(=O)NC1CC1)CC1CCCC1)C)OC C1(NC(C2CCCN(c3nccs3)C2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC12CC2 C(=O)(C(F)(F)C(F)(F)F)NCC1(F)CCN(C(c2ccc(OC)c(N)n2)=O)C1 N1(C(c2c(C)oc(CO)c2)=O)CCN(C(c2coc(CO)c2)=O)CCC1C C1(O)(CN(C(c2c(C)nc(C)[nH]2)=O)C)CCN(C(=O)CCc2ccncn2)CC1 C1(C)(CNC(C2CN(c3nnc(C(=O)OC)s3)CC2(C)C)=O)CC(C(C)C)=NO1 c1(C(N(C(CN(C(C(C)C2CC2)=O)C)C)C)=O)ccccc1C(F)(F)F C(CCCCC(=O)NCCCC(C)NC(=O)CCCN(C)N=O)(OC)OC CC1CCCCN1CCC(=O)NC1CC1CNC(C1CCC(=O)NC1)=O N1(C(C(COC(C)=O)C)=O)CCC(CO)(NC(c2coc(-c3ccsc3)c2)=O)CC1 N1(C(CCC=C)=O)CCC(O)(CCNC(C2(COC)CCCO2)=O)C1 C(=O)(CCC(C)CN(C)C)NC(C)CCN(C)C(c1cnn(C2CCC2)c1F)=O N1(CCNC(=O)NC2(C(F)(F)F)CCC2)CCCC(C(C)(C)C)C1=O CC1CN(C(c2csc(=NCc3ccn(C)n3)[nH]2)=O)CC(=O)N1 C#CCC(CC(=O)NCC1=C(Cl)CCC1)NC(=O)C(C)(C)C(=O)OC Cc1cccc(C(=O)NC2CN(Cc3cccnc3)CC2F)c1C c1(C(C)=O)cc(C(N2CC=CC2C(=O)NCC2COCC2O)=O)no1 N1(C(c2cccc(C)c2)=O)CCC2(CCCC2CNC(=O)C(=O)NC2CC2)CC1 O=C(C1=Cc2ccccc2OC1)NC1CCC12CN(C(=O)Cn1cnnc1O)C2 C1(NC(COC(CC)(C)C)=O)(CC)CCN(C(=O)CCCc2csc(C)n2)CC1 c1(-n2c(CCF)nc(CC(C)OC)n2)ccc2c(c1)OCO2 N1(C(CCCOCCC)=O)CCC(CC(N2CCC(C)(C)C2C)=O)C1(C)C C1(CNC(Cc2c(C)noc2Cl)=O)COCCN(C(c2ccc(N)cc2O)=O)C1 N1(C(CCCOCCOCC)=O)CC2(NC(C)=O)CCC1CC2.C1(=O)CN1 C1(NC(C2N(C(COC(CC)CC)=O)CC2)=O)CCN(C)C1(C)C c1(C(N2CC3(CCN(C(CC(C)OC)=O)C3)C2)=O)cnc2ncnn2c1N C12(NC(CSC)=O)CCN(C(c3cn4c(n3)SCC4)=O)CC1C2 N1(C(CSCc2cn(-c3n(C)ccn3)nn2)=O)CCC(F)(CNC(=O)CCF)C1.N c1(OC)cc2nc(C)cc(C(=O)NC(c3ccccc3)C(=O)NC)c2cc1OC c12coc(n1)C(=O)NCCOCCN2.c1(C2N(C(=O)OCC)CC2)ccccc1 CC1CCN(C(C2CC3(CSC3)C2)=O)CC1CNC(=O)CCc1cscn1 N1(C(C2N(C(C)=O)CCCC2)=O)CC2(CC2)CC1CNC(=O)Cc1cocn1 N1(C(C2CCC(=O)N2)=O)CC2(CC(NC(c3ncccc3Br)=O)CO2)C1 Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)C1=NOC(C)C1)C)S2 c1(OC)nc(C)ccc1C(N1CCC(CN(C)C)C1)C(=O)NC1CC(F)(F)C1 CCCCC(C(=O)NC(c1cn(C)nn1)C(=O)NC1CN(C)CC1O)N(C)C C1(C(=O)NCCc2ccncc2)CC2OCCC2N1C(=O)CCc1ccccc1 c1(OC)cc(C(N2CC3CC(NC(c4cnc(O)o4)=O)C2C3)=O)cc(N)c1OC C(=O)(C1OCCc2ccccc21)N(C(C)CNC(C12CC(C)(C1)OC2(C)C)=O)C c1(C(N2C(CCNC(C(F)=CC)=O)CCC2)=O)cnc(O)cc1OC C#CCCCC(C)C(=O)NCC1CN(C(=O)C2=C(C)OCC2)CC1(C)C c1(C(C)NC)cccc(C=O)c1.C1(N2CCCC2)(C(F)F)CCOCC1 Cc1c(F)ccc(C(=O)NCC2(C)CCCN(C(C3(C)CCCO3)=O)C2)c1N N1(C(C2CCN(C(c3n(CCC)ccc3)=O)C2)=O)CCN(C)C(CC)C1 c1(C(=O)NCC(CNC(CN(C(C)C)C)=O)CO)c(Cl)ccc(F)c1N c1(C(F)(F)F)cc(NC2CC(n3cccn3)C2)nc2ccccc12 N1(C(C2C3(CCN(C(C4CCN(C)CC4)=O)C3)C2)=O)CCCOC(C)(C)C1 CC(C)(CC(F)C(=O)NC1C2CCCCC12)NC(=O)CCS(N)(=O)=O C1(NC(=O)CC2(O)CCOC2)COCCC1CNC(=O)CCc1ccc(O)cc1 C1(N(c2nc(N(CC(CC)(C)OC)C)nc(C)c2)CC)CCc2cnn(C)c2C1 C1(CC(=O)N(C2CC2)CC2C(C)C2)CCC2(CC1)CCN(Cc1csnc1Cl)C2 C(=O)(C1CCc2cccc(O)c21)NCC1CN(C(c2c(C)nco2)=O)C(C)C1 c1(C(=O)NC2CCC(CCNC(COCCCC)=O)C2)cc2cccc(F)c2s1 CN1CCCC2(CCN(C(CC(F)C(C)(C)O)=O)C2)C1=O c1(C2C(NC(C(=O)NC3CC(C#C)C3)=O)C2)cccc(F)c1 C(=O)(CCCC(C)(F)F)NC(C1CN(C(c2cc(O)cc(O)n2)=O)CCO1)C N(C(=NCCC1CCCOC1)NC1CCC1)CC(CC)(C)C C1(c2n(C3(C)CC3)nnn2)(O)CCCCCCCC1.C12(CC1)CCNC2.CO C(=O)(C(O)CCCNC(=O)COCC(C)C)NC(CC)CC C1(C(N2C(CC)CC2)=O)C2CC3C(C2NC(C2CCC(O)CC2)=O)C13 C1(NC(CCCC(=O)NCC)=O)CN(C(=O)C(O)C(C)C)C2CCCCC12 CC(C)C(C(=O)N1CC(C)(NC(=O)Cc2cnnn2C)C1)c1cnn(C)c1 C1(CC(=O)NCC2(NC(c3cncc(C(N)=O)c3)=O)CC(=C)C2)CCOC1(C)C N1(C(C(C)OCC)=O)CCN(C(c2ccc(O)cc2CC)=O)CC1CC n1(CC(=O)NCC#CC(F)(F)F)cc(Br)cc(Cl)c1=O N1(C(C=Cc2occ(C)n2)=O)CC(C2CN(C(c3ncc4[nH]ncc4n3)=O)C2)C1 c1(C(=O)NC2CCC(CNC(c3c(C)c[nH]n3)=O)C2)c(C)sc2ccccc12 C(=O)(CCCNC(c1ocnc1C1CC1)=O)NCC(COCC)C C1(C(N(CCCOCCNC(C2C=CCCC2)=O)C)=O)CCCN(S(N)(=O)=O)C1 C(=O)(CC1COc2cc(O)ccc21)NC1(CNC(C2C(C)C2(F)F)=O)CCC1 c1(C(=O)NCCCCCNC(C(C)OCCC#C)=O)ccnc2cc[nH]c12 c1(-c2onc(Cc3ccc(OC(C)C)nc3)n2)ccc2c(c1)CCCNC2 C(=O)(C(COC)CC)NCCCN(C(c1c(CC)cc[nH]1)=O)CC1CC1 C1(C(=O)NCC(C)CNC(c2ccn(C(C)(C)C)n2)=O)CC(C)(C)CCO1 C#Cc1cc(C(N2CC(CNC(=O)CC(F)F)C(O)C2)=O)ccc1Cl c1(CCC(=O)NC(CC=C)CNC(C2(C(=O)OC)CC2)=O)ccnc(Cl)c1 C1(CNC(CN(C(=O)C=CS(C)=O)CCC#C)=O)CC2CCC1C2 Cc1cc(C(=O)NCC2(C)CCCN2C(=O)COc2ccc(Cl)cc2)cc(O)n1 C1(C(N2C(CCNC(C3C(C)=CCS3)=O)CCC2)=O)CCN(CC(F)F)CC1 C(C(=O)NC(C)Cc1cccnc1)(C(C)(C)O)NC(C1(C(=O)OC)CC1)=O N1(C(c2cc(C)sc2)=O)CCC2(CCC2)C(CNC(c2cc(F)cc(F)c2)=O)C1 c1(CN2C(=O)CCN(C(c3ccc(Cl)s3)COC)C2=O)cc2cccnc2[nH]1 c1(C(=O)NC(CNC(C(C)=C2CC2)=O)C2CC2)ccc(C2CCCN(C)C2)cc1 C1(C#N)(C(=O)NCC2CCC(NC(CN3CCN(C)CC3)=O)CC2)CC2CC2C1 C(C(CC(C)C)C(=O)NCC1(C(=O)NCCC(CO)C(C)C)CCCCC1)OC c1(C(=O)NC2(CO)CCN(C(C(C)C3CCC3)=O)C2)cccn(C2CC2)c1=O C=CCC(CC)C(=O)N(CC(C)CNC(=O)CSc1ccccc1C)C N1(C(C2(C(=O)OCC)CC=CC2)=O)CC2CC(C1)N(C(=O)CC1(N(C)C)CC1)C2 N1(C(C2CC(OC)C2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1c1nccn1C N1(C(CC(=O)NCC#C)=O)CCC(CC)(NC(C2NC(=O)OC2C)=O)CC1 CCCC(CCC)C(=O)NC1CCCC12CN(C(=O)C(CC)n1ccnc1)C2 N1(C(C2C(=C)C2)=O)CCCCC1CCNC(=O)C(c1cccc(C)c1)=O CCC(CN(C)C)CC(=O)N1CC(CO)(NC(c2cccc(CO)c2C)=O)C1 c1(C(=O)NCC2C(NC(C=Cc3n(CC)ccn3)=O)CC2)ccc(OC)c(O)c1 CS(=O)(=O)c1ccc(CN(C2C(c3ccccc3)CNC2)C2CC2)cc1 N1(C(c2[nH]cc(CC)n2)=O)CCCCCC1C(N1CC2CCCC2C1)=O CCC(CCC(=O)NC1CCCCCC1O)NC(C1OC2CCC1C2)=O C1(C(=O)NC2(C(F)F)CCN(Cc3ccccc3)CC2)Cc2cccnc2C1 N1(C(=O)NC(c2c(OC)cccc2)C)CCN(c2ncccn2)CC1C c1(C(=O)NC2C=CC(CNC(=O)C=CC(F)(F)F)C2)cc2n(n1)CCCC2 C(=O)(C(C)CCCC(C)=O)NCC1(CC(N2CC(C#C)C(O)C2)=O)CC1 C#Cc1ccc(C(=O)N(CC(=O)NCC=C)CC(C)C)cc1 c1(C(N2CC(N(C(CC(C(C)C)O)=O)C)C2)=O)cnc2[nH]nc(O)c2c1 C1(NC(C(C)N(C(C2C3CCC(C3)C2C)=O)CC)=O)CN(C)C(=O)C12CC2 C(=O)(C(F)CC(C)(C)NC(=O)C#CC1CCOC1)NCC1CC(C(=O)OC)C1 C1(NC(C2CN(CC)C(=O)C2)=O)CCN(Cc2cncs2)CC1O C1(C)(C(=O)NC(C2(C(=O)NCCC(=O)OC)CC2)C)CCOC(C)C1 c1(C(N(CC(C)NC(=O)CC2(O)CCCC2)C)=O)cn(CCO)nn1 C1(C(=O)NCc2ccc(C)cc2)CC(F)(F)CN1Cc1cnc(Cl)cc1Br C(C(CC(C)C)C(=O)OC(C)(C)C)NCc1ccc(CCCCC)cc1 Cc1cccc(F)c1C(=O)NCC1CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CCO1 C1(CCC)(C(N2CCC(N(CCO)C(C3CCC(C)(C)O3)=O)C2)=O)CCNC1=O Cc1nc(O)ccc1C(=O)NCC(CC1CC1)C(=O)NC(C)C(=O)N(C)C N1(C(CC(c2ccc(Cl)cc2)C)=O)CCOC2CNCCC12 Cc1cnc(C(C)NC(c2cc(C3CC3)cs2)c2nnnn2CC2CC2)s1 c1(C(N2CCC(CSC)C2)C(=O)NC2CC(N3CCC3)C2)cc(F)ncc1F CCCCC(C)CCC(=O)NC1C2CC(NC(c3csc(C4CC4)n3)=O)CC12 C1(C(=O)NC(C)(CO)C(=O)NCC2CC3CCC2O3)CCC2(CC1)CC2 c1(C(=O)NCCC(C)N(C(=O)CC2CC2)C)nccc2c1[nH]c1ccccc21 C1(NC(c2c(COC)cccc2)=O)CN(C(C2(C)CCCO2)=O)CC(F)(F)C1 C1(C(=O)NC(C(=O)OCCC)C)CN(C(C2(F)CCC2)=O)CCO1 c1cnc(C(=O)NCCOCCN(C)C(c2ncnn2CC)=O)c(Cl)c1.CCSC n1(CC)nc(C(=O)NC(C(N2CCOCC2CO)=O)c2ccco2)cc1C C=C1CC2CCCC(C1)N2C(=O)CC(C1CC1)NC(=O)CCc1noc(C)n1 N1(CC2CCC(C)(C)C2)C(=O)CN(CCC2(C)CC2(F)Cl)C1=O C(=O)(C1CCCc2sc(=N)[nH]c21)NCCNC(C1(C)CC1(F)F)=O CC1CCN(C(=O)Cc2cncnc2)C1CNC(c1ccc(-c2ccco2)o1)=O N1(C(C(C)Oc2cccc(F)c2)=O)CCC(NC(=O)C2=CCCS2)C12CCC2 c1(OC(C)C)cccnc1N1CCN(C(C)C(=O)NCC(=O)NC(C)C)CC1 C1(COC)CN(C(c2nnc(S)n2C)=O)CCN1C(=O)CSc1ccc(C)s1 CCS(=O)(=O)C1(CS(=O)(=O)c2cccs2)CC1.C1C(=O)OC(=O)CN1 Cc1nc2cc(C(=O)NCC3(C)CC(NC(C4CC=CCC4)=O)C3)cnc2s1 C12CCCCN(C1)C2.C(=O)(COCCOCCOCCO)OC c1(C(C(N2CCC(N(C(=O)Cc3cscn3)CC)C2)=O)(F)F)ccc(C)cc1 C1(C(C(=O)NCC(CC)CO)(C)C)CCCN(C(=O)C(O)CCSC)C1 CCCCCCCC(F)C(=O)NC(C)(CNC(c1conc1C)=O)CO N1(C(C(N(C(C(C)NC(=O)C2CC2)=O)C)C2CC2)=O)CCC2(CCSC2)C1 N1(C(c2cncc(C#C)c2)=O)CCCCC(N=c2[nH]c(Cl)ncc2[N+](=O)[O-])C1 N1(C(c2n[nH]c(C)c2F)=O)CCC2(CCCN(C(=O)CN3CCN(C)CC3)C2)C1 N1(C(C(c2ccccc2)SC)=O)CCC(CCNC(=O)C2=CCSC2)C(F)(F)C1 N1(C(c2c(C)nc(O)cc2)=O)CCCC(C)(C)C1CNC(C1(CO)CCCO1)=O c1(CNC(CC2N(C(CSC)=O)CCC2)=O)cccc(O)c1F c1(CN2C3CC(CNC(COCC)=O)C2CC3)nc2ccc(OC)nc2s1 c1(C(=O)NC(CN(C(CC2N(CC)CCC2)=O)C)C)ccc(F)cc1C1CC1 C1(NC(COCCC=C)=O)CCCC12CCN(C(=O)C(N1CCSCC1)C)CC2 Cc1ccc2c(c1)SC(C(=O)NC1CC(NC(c3coc(O)n3)=O)CC1O)C2 C(=O)(CC(C)CC(C)C)N1C(CNC(c2nccc(OC)c2C)=O)C(O)C(O)C1 N1(C(C2CC(CC)C2)=O)CC(C(=O)NCC2(CC)CCC2)(CC)C1 N1(C(C(CC)(C)CNC(=O)C(F)F)=O)CCC2CC1C(=O)O2 N1(C(CC)=O)CCCC12CCN(C(=O)CCC(=O)OC)C2.C12CCN(C1)C(=O)C2 c1(CNC(c2n(C(CC)C)nnn2)c2coc(C)n2)cccc(Br)c1 S(=O)(=O)(c1ccc(NCC(O)CC2CCC2)c(C#N)c1)NCc1c(CC)nn(C)c1 c1(CC(=O)NCCC2(OC)CN(C(c3sc(CO)nc3C)=O)C2)ccc(C)cc1 N1(C(c2n(C)c(S)nc2)=O)CCC(C2(NC(=O)CC3CC=CCC3)CC2)CC1 Cc1ncn(C)c1C(=O)NC(C)C(C(C)C)NC(c1cnn(CC2CCC2)c1)=O N1(C(c2cc(C)ns2)=O)CC(CNC(=O)CSCc2csc(=N)[nH]2)CCC1C N1(c2c(C)cncn2)CC2(C1)C(NC(C1CC3C(C1)C3(C)C)=O)CCS2(=O)=O C1(CCNC(C2C=CCC2)=O)CN(C(=O)C(F)=C2CCC2)CCCO1 C1(NC(c2c(OC)noc2C)=O)CCN(CCCOC(C)C)CC1O.C1C(=O)O1 C(=O)(C(C)CC(C)C(C)=O)NC(CCC)C(O)C(=O)NC1CC(C)(OC)C1(C)C c1(C(N(CCN(C)C(C2CSCCS2)=O)C)=O)cnc(N(C)C)s1 N1(C(C2CC(C)(NC(C3COCCO3)=O)C2)=O)CC2(CC(CO)CO2)C1 C1(NC(c2c(CC)oc(C)c2)=O)CC(C(=O)NC(c2cccnc2C)C)=CC1O C1(C(=O)NCC(COC)F)CC=CCC1CSC C(=O)(C(CC)NC(=O)Cn1cc(CC)cn1)N(CC(=O)N(CC)CC)C c1(-c2cc(F)cc(F)c2)cc2c(s1)CCN(C(=O)CCC(C)=O)C2.C(=O)NCC c1(-c2c(-c3n(-c4n(CC)ccn4)ccn3)csc2)cccnc1-c1ccns1 N1(CCC)CCN(C(C2CCC(c3cccc(Cl)c3)CC2)=O)CC1 C(=O)(CC(O)CNC(=O)C(C)(C)OC(C)C)N1C(C(=O)OC)CC1C C1(CNC(C2C(C(=O)OC)C2)=O)CCC(NC(c2ccon2)=O)CC1 c1(C(=O)NC(COCC)C(=O)NC2CC3C=CC2C3)cc(S(N)(=O)=O)cs1 c1(OC)cc(OC)c(NC(C2CN(C(=O)CCc3ccc(C)s3)CCN2)=O)cn1 C(C(C)(C)C(C)(C)C)NC(C(CSCC)N(C(=O)CC(C)(C)SC)C)=O c1(C(=O)NCCC(C)NC(c2c(CC)cccn2)=O)oc2ccccc2c1C Cn1nnnc1SCC(=O)NC1(CCNC(C2CC2C(F)F)=O)CC1 c1(C(=O)NCCN(C(CC=C)C(=O)NC)C2CC2)ccc(OC)nc1C CCCCC(CC)C(=O)NCCCOCCN(C)C(C1CSCCS1)=O C(CS(=O)(=O)CC(=O)N1CCN(C(c2cnn(C)c(=O)c2)=O)CC1CCO)OC c1(C(N(CCC)CCNC(=O)C(c2ccnn2C)O)=O)cc(Cl)cc(F)c1N c1(C(=O)NC2CC(C)N(C(c3cncn3C)=O)C2)cc2c(Cl)cccc2s1 N1(C(C(C)OCOC)=O)CCC2(CCC2)C(C(=O)OC)C1.O(CP(C)(C)=O)CC(=O)NC C#Cc1ccc(Cl)c(C(=O)NC(C)CN(C)C(c2cc(C(CC)CC)no2)=O)c1 Cc1cc(F)ncc1C(=O)NC(C1CCN(C(=O)CCc2cccs2)C1)C c1(C(C)C)sc(Cl)nc1NC(N1CCN(C)CC1)=O.C(=O)(C(=O)NC)NCCC(N)=O C(C(F)(F)C(F)(F)F)OCCC(=O)NCC1(C(C)NC(C(CC)SC)=O)CC1 Cc1cc(Cl)cc(N)c1C(=O)NC1CN(C(=O)CCN2CCCC2)C(C)(C)C1 C1(NC(=O)CCCc2cncs2)CC2CN(C(=O)CCCCC3CCCCC3)CC12 Cc1ccc(CC(C)NC(=O)NCc2cc(C)ncn2)nc1 c1(C(N2CCC(C)C(NC(C3(F)CCCC3)=O)C2)=O)cc2ccccc2o1 C(C(=O)NC(c1cc(Cl)cc(Cl)c1)CC(F)(F)F)(C(C)C)(C(C)C)NC(C)=O C1(=CC(=O)NC2CC23CC(NC(c2n[nH]cc2Br)=O)C3)CN2CCC1CC2 C1(NC(C(C)CC(F)(F)F)=O)CCCCC12CCN(c1nnc(C3CC3)s1)C2 C1(CN(C(C=CC)=O)C)CN(C(c2cccc(C3CC3)c2)=O)CCO1 Cc1cccc(Br)c1OCC(N1CCC(C(C)NC(c2ccns2)=O)C1)=O C1(CNC(c2ccc(F)o2)=O)CC2(CCN(C(c3cc[nH]c3C3CC3)=O)C2)CO1 N1(C(c2ccc(F)c(CO)c2)=O)CC2CCCN(C(C3C4CCC3CC4)=O)C2C1 C(=O)(C1CCCn2nccc21)N1CCCCC(N(C(=O)C2=COCC2)C)C1 c1(C(=O)NCC(C)CNC(=O)CN(c2ccccc2)C)c(O)ncc2c1CCC2 C1(NC(Cc2ccc(C)nc2Cl)=O)CN(C(=O)Cc2ccsc2)CCC1(C)C c1(C(=O)NC(CC)CNC(c2cncc(F)c2Cl)=O)ccn(C)c(=O)c1O Cc1ccnnc1C(=O)N(C1CCN(C(=O)Cc2ccccc2F)C1)C N1(CC(=O)NC(C2CC2)C2CC2)CCCC(O)C1.C(CCl)O C(=O)(CCCCn1cc(CCC(=O)OC)nn1)N(CCCOC)C(C)C c1(N(C)C)ccc2cc(C(N3CCN(C(=O)Cc4cncs4)CC3)=O)ccc2c1 CCCCC(O)C(=O)NC(CNC(=O)CCCCSC)CC(F)(F)F C1(NC(CC(C)c2cnn(C)c2)=O)CC2CN(C(=O)C(C)(C)C#N)CC2C1 c1(OC)ccc(Cl)c(C(=O)NCCC2CCN(C(=O)C3=COCC3)C(C)C2)c1 c1(CC(=O)NCC(CNC(CCCOC)=O)F)c[nH]c2cccnc12 c1(C(=O)NCC2CCC(C(=O)NCc3cc(CC)no3)C2)cc(C)n(C)c1 c1(NCC2(C(C)N)CC2)ccc(S(=O)(=O)NCCCc2ccccc2)cc1Cl Cc1cc(C(=O)NC(C2CN(C(=O)CC3CC4(CC4)C3)C2)C)ccc1N n1(CC(=O)NC(COCC(C)Oc2c(OC)cccc2)=O)cnc2c1CCCC2 CCCC(C(O)C(=O)NC1CCC1COC)NC(=O)CC1=CCCC1 C(=O)(C(O)C(C)(C)C)NCCN(CCCN(C)C)C(=O)Cn1nnc(C2CC2)n1 N1(C(CCNC(C)=O)=O)CCC(C(N2CCN(C(C)(C)C)CC2)=O)C(O)C1 CC(CO)(CO)C(=O)N1CCC2(CC2C(=O)Nc2nc(Br)cn2C)C1 O=C1OCc2c(C(=O)NC3CC(O)CN(C(=O)CCCC(F)F)C3)cccc21 N1(C(C2COC(C)(C)OC2)C(=O)NC2(C)CC2)CCCC(C)C1C1CCC1 CN1CCOCC1C(=O)NC1CCC(C(=O)NOCC2(C)CCC2)C1 Cc1nc(C)c(C(=O)N(CCCCCNC(c2cnc(C(C)(C)C)o2)=O)C)[nH]1 c1(NC(C2(OC)CCN(C(c3ccc(C4CC4)s3)=O)C2)=O)ccc(Cl)c(C)c1N CCC(O)C(F)(F)C(=O)NC1CCN(C(=O)CC=Cc2ccccc2)C(C)C1 c1(OC)ccncc1CNC(=O)C(CC1CCCC1)NC(=O)CN(C)C C1(F)(CNC(C2C=CCC2)=O)COCCN(C(=O)CC2CCCCC2)C1 c1(C(=O)NCC(C)CNC(c2cc(Cl)ccn2)=O)cc(O)nc2c1CCCC2 C(=O)(C(CC#CC)NC(c1ccc(C)cc1O)=O)NC(C=C)(C)C C1(C(=O)OCC)COCCN(CC(N2CCOCC2)C)C1 CC1(C)OC(=O)CC1C(N1CCOC(CC(=O)NOCCC2CC2)C1)=O c1(C(=O)NCC2C(NC(C3CC(=O)NC(=O)N3)=O)CCCC2)cc2cccnn2n1 C1(NC(C2(SCC)CC2)=O)COC2(CCN(C(=O)CCC3CCC3)C2)C1 c1(C(=O)NCC2CCN(C(c3ccc(SC)cc3)=O)C2)cccc2c(C)[nH]nc12 N1(C(CCNC(=O)OC)=O)CCOCC(C(=O)Nc2cc(C)ccc2C)C1 Cc1cnc2c(C(=O)NC3CC3NC(C3Cc4cc(F)ccc4O3)=O)cnn2c1 C=CCC(CC)C(=O)NCC(O)C(=O)Nc1cnccc1OC C(=O)(C(CC(C)C)CC(C)C)N(CCCCCNC(Cc1ncc(C)o1)=O)C Cc1c(C(=O)NCCN(CC(C)O)C(c2coc(Cl)n2)=O)oc2ccc(Cl)cc12 c1(C(=O)NCC(CNC(CCCCOC)=O)O)ccc(=O)n(CCO)c1 C1(C(N2CCCC(CN(C)C(C3(CCF)CCC3)=O)C2)=O)CC2(C1)CC2(F)F C(=O)(C1=NOC(C)C1)NC(C(=O)NCC1ON=C(CC)C1)Cc1ccoc1 S(=O)(=O)(c1[nH]c(=NCC2C=CCC2)ccc1Br)NC1C(C)(N(C)C)CCC1 C(=O)(C1CCc2ccc(Cl)nc21)NC1C(CNC(C2=C(C)OCC2)=O)COC1 Cc1sc(O)nc1C(=O)NC1CC=CCC1NC(C1(N2CCCC2)CCC1)=O Cn1cc2c(C(=O)NCC3C4CN(C(c5nscc5N)=O)CC34)cccc2n1 c1(CNC(C2CC2CNc2cc(C(F)(F)F)cc(O)c2)=O)cc(Cl)cc(Cl)c1O C1(C(=O)NC(CC#C)(C)C)CC(C)CN1C(=O)CCSCC C(c1cccnc1)=CC(=O)NCC(CO)NC(C(n1ncc(C)c1)C)=O c1(CC)cccc(CN2CC(c3ccsc3)CC2C)n1 C1(C(=O)NCC2(OC)CCN(C(=O)C(C)(C)CCC#N)C2)CC2C=CC1C21CC1 c1(C(N)=O)c(F)ccc(NNC(=O)NCCCn2ccnc2)c1C C1(C(=O)NC(C(=O)NCCC(=O)NCC#C)(C)C)CCCNC1=O CC1(NC(C2CCC(OC(F)F)CC2)=O)CCCN(C(=O)C=Cc2ccco2)C1 C#Cc1cc(C(=O)NCC(CO)NC(c2ccc(O)nc2)=O)cc(F)c1 N1(C(C2(CC)CCC2)=O)CCC(NC(c2cc(C(F)F)cnc2OC)=O)C(F)C1 CC(C)CCC(=O)NCC12CC(NC(c3ccc(C(=O)OC(C)C)nc3)=O)(CO1)C2 N1(C(CCCC=C)=O)CC2CCC1CN2C(=O)CNc1ccc(C)cc1 N1(C(N2CCCc3occc3C2)=O)CC(O)CC2CCCCC12 C1(NC(CC2C=CC(NC(CCC3CCC(C)O3)=O)C2)=O)CCOCC1(C)C O=C(N1CC2COCC2O1)c1ccc2c(Br)[nH]nc2n1 c1(C(=O)NCC2OCCCN(C(CC(C)C)=O)C2)cnc2cnccc2c1 C1(NC(c2[nH]c(CC)c(Cl)n2)=O)CCN(C(c2ccc(F)c(F)c2)=O)C1(C)C Cc1cc2ccc(C(N3CC4CC4(NC(c4n[nH]c(C)c4C)=O)C3)=O)cn2c1 c1(N(CC(C)CNC(c2ccsc2)=O)C)cc(-c2ccccc2)ncn1 c1(C(=O)NCCC2(O)CCN(C(c3c(CCC)n[nH]c3)=O)C2)cc2c(s1)CCC2 c1(OC)ccc(Cl)c(CNC(C2(c3nccs3)CCCCC2)=O)n1 CCC(CC(C)C)C(=O)N1CCC(CN(c2nccc(C#N)n2)C)C1 c1(C(N2CC(C)(NC(C3CCCC(N(C)C)C3)=O)C2)=O)cnc2cccnn12 n1(CC(N2CC(CNC(C3C4COCC34)=O)OCC2)=O)cnc2sccc2c1=O C1(CC)CC(C(=O)NCC2CCC(F)(F)C2)CCN1C(C1CC(C)=NO1)=O C1(NC(CC)=O)CCCN(C(=O)Nc2cccc(-c3ccccc3Br)c2)C1 CC1CN(C(=O)CCNC(C2CCC2)=O)CCN1C(c1cn(C)nc1Cl)=O c1(OC)cc(C)sc1C(=O)NC1(CNC(=O)COc2cccc(F)n2)CC1 C(CN=c1[nH]c(=NC(C)C2CC=CCC2)[nH]c2ccsc12)N(CC)CC C#Cc1cc(C(N2CCC2CNC(=O)CN2CCCS2(=O)=O)=O)ccc1C C1(C2CCN(C(C3CC4(CCCO4)C3)=O)C2)(NC(=O)CC2(CO)CC2)CC1 c1(N2CC(C)=C(C)C2)nc(N2CCCC(CO)C2)nc2cccnc12 CC1CCC(C(=O)NCC(O)CCO)CN1C(=O)Cc1cccnc1O C1(NC(C2CSCCS2)=O)CN(C(c2ncncc2Cl)=O)CCC1CO C(=O)(C(CC(C)C)OC)N1CC(CCC=C)(C(=O)NCCC=C(C)C)C1 N1(C(c2cc(OCC)n[nH]2)=O)CC2CC1CCN2C(=O)CC1=CCCCC1 C1(C)(CC)C=C(C(=O)N(CCNC(c2ccc[n+]([O-])c2)=O)C2CC2)C1 C1(C(N2CCN(C(CC=C)=O)C(CS(C)(=O)=O)C2)=O)CC2(C1)NC(=O)NC2=O Cc1cc(NC(=O)CCC2CCCN2C(=O)C(C)S(N)(=O)=O)cc(C)c1F C1(CCNC(C(C)CN(C)C)=O)CCCCN1C(=O)CCCCc1ccccc1 N1(C(CN(C(C)=O)C)=O)CCCCC(N(C(=O)C=C(C2CC2)C2CC2)C)C1 C(C(COC)C(=O)NCC1(c2ccccc2)CC1)NC(C1CC(=C)C1)=O C1(N(C(=O)CSCc2ccccc2)C)CCCC(NC(c2cn(CC)cn2)=O)C1 C(=O)(CC(F)(F)C(F)F)N(C)CC1CCCCN1C(C12CCC(CO)(CC1)C2)=O C1(NC(c2cc(F)c(Br)cc2F)=O)CCCCCN(C(C2(C3CC3)CC2)=O)C1 c1(C(N2C(C)CCN(C(C(C)=C3CCC3)=O)C2)=O)cc(F)c(F)c(N)c1Cl c1(NC(c2n(CCCOC)nnn2)C(C)COCC(C)C)c(F)cccc1Cl c1(C(N2CC(NC(CC3(C)CCC3)=O)C2)=O)cccn2nncc12 S(=O)(=O)(c1cncc(Cl)c1)Nc1nc(C#N)c(Br)cc1 c1(C(=O)OCC)cnc2ccc(CN3CCC4(C3)CNC4)cn12 S(=O)(=O)(c1cc(Cl)c(F)cc1F)N1CC(C)OC(C(=O)O)C1C N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CC2CCCC2(CNC(C2CC2)=O)C1 CCCC(O)C(=O)N1CC(C(=O)NC2CCO2)(COC)C1 c1(C(N2C(CCCNC(c3c(C)cn(C)c3)=O)CCC2)=O)cc(O)ccc1N c1(C(C)OC(=O)Cc2csc(-c3cnn(C)c3)n2)ccc2c(c1)OCCO2 c1(CC)cc(C(=O)NCCC2CN(C(C3CC34CCOC4)=O)C2)nn1C C(=O)(N=c1ccn(C2CC2)[nH]1)C1C(=O)N1.c1(C(=O)O)[nH]nnc1CO CN(C)S(=O)(=O)N(C)CC(N1CC2(CC(NC(C3CCC(C)(F)CC3)=O)C2)C1)=O N1(C(C(C2CC2)OCC)=O)CCN(C)C(CNC(=O)C=Cc2cc(OC)ns2)C1 C(N=c1[nH]cnc(C)c1OC)C1CCC(NC(c2ccc(OC)cc2)=O)C1 C(CC(C(=O)N1CC(OC(C)C)C1)NC(C12COCC1C2)=O)OC c1(C(=O)CNCCC(F)(F)F)ncn2c1CCC2.C1CC1 N1(C(C(=O)NC(C)C)=O)CC(C)(C)OCC1CNC(c1ccc(F)c(F)c1F)=O N1(C(C=CC(C)C)=O)CCN2CCN(C(C3(c4ncco4)CC3)=O)CC2C1 N1(C(c2c(CNC(C(CCC)OCC)=O)noc2)=O)CCOC(C)C1CO c1(CC(=O)NC2CN(C(CCOCC)=O)C2)ccc(F)cc1F n1(CC)ncc(C(=O)Nc2cccc(NC(=O)C(C)(C3CC3)OC)c2)c1C1CC1 c1cc(N2CCOCC2)c2c(c1)CCN(N1CCOCC1CO)C2 c1(CSCC(=O)N(CC(C)(C)NC(CC2C(C)CCO2)=O)C)ccc(Cl)nc1 C(=O)(C1CCCn2cncc21)N1CCC(NC(C(C)n2cnnn2)=O)CC1 N12CC3CC(CC1C3)NC(=O)C2C.c1(C(=O)NC(CC)C)ncccn1 c1(CNC(=O)C(=O)Nc2ccccc2)ccc[n+]([O-])c1.C12(F)CC(C1)CNC2=O CC(CC(=O)N1CC(O)CC1CC(=O)NCc1ccc(O)cc1F)C(F)(F)F C1(CCC(=O)NC2(C(F)(F)F)CC(=C)C2)CCCCN1C(=O)C(C)SCCCC C#CCCCCCNC(=O)CC1(C)CCN(C(=O)C(C)(C)N(C)C)C1 C12(C(N3CC(C(C(=O)NCCCP(C)(C)=O)OC)C3)=O)CCC(C1)C2(C)C C1(C(N2CCC(C(=O)NCC(C(=O)NC)C)C2)=O)COCC(C)O1 Cc1cccc(CC(N2CC(C3CCCCN3C(=O)CNC(N)=O)C2)=O)c1 Cc1cc(C(=O)NC(C(=O)N(c2cccc(Cl)c2)C)C(C)C)nn1C c1(C(=O)NCC2CC(F)(CNC(C3CC34CCOCC4)=O)C2)cccc(F)c1O C(=O)(C1=CC2CC=CCC12)NC1CN(N2CCC(C(=O)OC)CC2)C1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2(SC)CCC2)=O)CCCO1 C(=O)(CCC(F)(F)C(F)F)NC(c1ccc(C)cc1)CNC(=O)Cn1cncn1 C(=O)(CCC(=O)N(C)CC1CCN(C(C2CCS(=O)CC2)=O)CC1)OC C1(C(=O)NCC2OCCN(C(c3cccc(CC)n3)=O)C2)CCCCNC1=O N1(C(C2CC2NCc2ccc(C(F)(F)F)cn2)=O)C2CCC1COC2 C1(NC(C2COCCN2c2ccccn2)=O)CC(O)C(O)C1O N1(C(C2(C)N(C(CC3C(C)OCC3)=O)CC=C2)=O)CCC12CN(C)C2 C1(c2cn(CCC(C3CCCC3)OC)nn2)CCCCC(=O)C1 Cc1cc(Cl)c(C(=O)NC2CC(NC(=O)CCOCC3CCC3)CC2O)s1 C(=O)(C(C)C(C)(C)C)NC1(C(N(C)CC2C(C)COCC2)=O)CCSC1 c1(NC)ccccc1C.CCCCCCNC(C)C(=O)NCCNC(C1CC(OC)C1)=O c1(CNC(C2CC(O)(CNC(C(C)=C3CCC3)=O)C2)=O)cc(C)cc(F)c1 CS(=N)(=O)c1ccc2c(c1)N(C(=O)Cc1cnoc1)CC2 c1(OC)c(C(=O)NC2CC3(CCCCO3)C2)cc(C)c(Br)c1F N1(C(C(CC(F)F)NC(c2n(C=C)nnc2)=O)=O)CCN(C)CC(O)C1 C1(C(N2CCC(N(CC(C)C)C(C3(C)CC3(F)F)=O)CC2)=O)CCOCC1(C)C c1(C(=O)NCC(C)N(CCOCC)CC)ncnn1-c1ccccc1 N1(C(c2c(CC)ccs2)=O)CCC(C)(CCNC(=O)CC(C)C2CCC2)CC1 C1(O)(CC)CCN(C(=O)CCCC(C)NC(c2cnc(O)o2)=O)CC1 C(=O)(C(F)(F)C(O)C1CC1)NC1CC(N(C(c2ncn(CC)c2)=O)C)C1 C1(O)(CN(C(=O)C(F)(F)C(F)F)C)CCN(C(c2cccc(N)c2O)=O)CC1 CCCCC(CC(=O)NC1CCCCCC1O)NC(C1CCC2(CCC2)O1)=O c1(NCC(C)CNC(=O)CSc2cccs2)snc(Cl)c1C#N CC(C(C)(C)C)=CC(=O)NC1CC1NC(c1cc(-c2ccccc2)sn1)=O C(CC)(C(=O)N1CCC(CCC(=O)N(C2(COC)CCC2)C)C1)OCC c1(CNC(=O)NCC=CCC)cc(F)ccc1O CCC(O)C(F)(F)C(=O)N1CC=C(C(=O)NCc2ccc(CO)cc2)CC1 c1(C(N2CC=CC(NC(c3cc(C)c(C)nn3)=O)C2)=O)cc2ccc(F)cc2s1 C1(C(=O)NCC2C(NC(c3cn(C(C)(C)C)nn3)=O)CCC2)CC2(C1)CC2(F)F C1(CNC(C(C=C)(F)F)=O)CC2CCCC2N1C(=O)CCc1cnc(C)o1 C1(NC(c2nc(C)c(C)s2)=O)CC(C(=O)NCC2CCOC2(C)C)C12CCC2 N1(C(C2(C#C)CCCC2)=O)CCN(C(=O)CC2(CO)CC2)C(COC)C1 CC#CCC(C(=O)NC1CCOC(C)C1)NC(C1CNC(=O)O1)=O c1(C(N(C2CCC(NC(c3cnn[nH]3)=O)C2)C)=O)noc2ccc(Cl)cc12 C1(C(=O)NCC2CCN(C(=O)C(c3ccc(F)cc3)F)C2)CCc2nn[nH]c2C1 C1(C(CC)CC)CN(c2cc(NC(c3cccnn3)C)ncn2)CCO1 n1(CC(=O)NC2(C)CCN(C(C3(C#C)CC3)=O)C2)cnc2ccc(F)cc2c1=O c1(CC(C)C(=O)NC2CN(C(c3ccc(C4CC4)o3)=O)CC2F)ccccc1Cl c1(CNC(CN(CC#C)C(c2cnsc2C)=O)=O)cn(C)nn1 C1(OCCCN(C(=O)Cn2ccnn2)C)CCN(C(C2C3CCN2CC3)=O)CC1 C1(NC(C(C)SC(C)C)=O)C2CCCN(C(c3ccns3)=O)C2C1(C)C C(=O)(C(CCC(C)C)NC(c1cncc(NC)c1)=O)N1CC(CCC)OCC1 C(C(C)(O)C(=O)NCC1CCCN(C(=O)CC2CC(C)=NO2)C1)OC c1(NC(C2C3CN(C(c4c(C)c(Br)cnc4)=O)C2C3)=O)cc(C#N)ccc1F c1(C(=O)NC(CNC(C(CC)C)=O)C)cccc(OCCCOC)c1 N1(C(CNC(=O)OC)=O)CCC(N(C)C(c2ccnc(OC)n2)=O)C(C)C1 C(N=C(NCC(F)F)NC1CC1c1cccc(Cl)c1)C1C(c2cnn(C)n2)C1 N1(C(CC(=O)NCC)=O)CCN(C(C2C=CCC2)=O)C(=Cc2ccccc2)C1 C(CC(C(=O)NCC(C(F)(F)F)c1ccon1)NC(=O)OC(C)(C)C)OC N1(C(C2CC3CC2C3)=O)CCCC(C2CCN(c3ncc4ncnc-4[nH]3)C2)C1 O=C(CCCCN1CCC1)NCC1CC(NC(c2sccc2CO)=O)C1 n1(CC)nnc2c1C(C(=O)Nc1ncccc1C)CN(C(c1ccncn1)=O)C2 C(CC(O)C(=O)NCC(C1CCCC1)NC(=O)CN1CCC(CO)CC1)N(C)C CC(C)CN(Cc1ccccc1)N(CCN1CCCC1=O)C(C)CO N1(C(c2ccc(OC)cc2Cl)=O)CC2CC1CN(C(c1cc(Br)c(C)o1)=O)C2 CCCC(CC)C(=O)NCC1CC(C)(NC(c2ccc(N(C)C)nc2)=O)C1 N1(C(C(CC(=O)OCC)C)=O)CCC2(CCC(NC(=O)CN(C)CC)C2)CC1 Cc1cn2ccnc(C(=O)NCC3CCCN(C(=O)C(C)C4(O)CCC4)C3)c2n1 C1(C)(C(=O)NCCCCNC(C2CCC(C)O2)=O)COC(=O)C1 C1(C(N2CC(O)(CCNC(CCSCC(N)=O)=O)C2)=O)CC2(CC2)CN1C N1(C(CCCC#N)=O)C2CCC1CN(C(C13CC(c4cccnc4)(C1)C3)=O)C2 N(C1CCC(=O)c2ccccc21)C(=O)C1=NOC2COCC12 Cc1nc(C(=O)NCC2C3CN(C(C4(N(C)C)CC4)=O)CC23)c(C)n1C1CC1 C1(C(=O)NC(CO)CCO)CC2CC1CC2NC(c1cc[nH]c1)=O Cc1cc(CC(=O)NC2(CNC(=O)C(C)SC(C)C)CC2)ccc1F C#Cc1ccc(C(=O)NC2C3CN(C(=O)CCC(=O)c4cccnc4)CC23)nc1 c1(C(=O)NC(CNC(c2c(NC)cnnc2)=O)(C)C(C)C)cnccc1C#N c1(C(=O)NC2CC(NC(C(C)SC(C)C)=O)C2)cscc1C(C)C C1(C(=O)NCC2(N(C)C)CN(C(=O)C(C)SC)C2)COCC1(C)C.CO N1(C(CC2(NC(C)=O)CC2)=O)CCC(NC(=O)C(C)(F)C(C)(C)F)C(CO)CC1 N1(C(CCCCCSC)=O)CC(=O)N2CCOCC2(CNC(C2CCCS2)=O)C1 C(C#Cc1ccccc1F)NC1C(O)CCCC1c1ccc(F)cc1 N1(C(CN(C)C)=O)CC(NC(=O)C(c2ccc(O)cc2)(C)C)C(n2cccn2)C1 C(C)(C)(CCCC(=O)NCCC(C)SC)NC(C1CCC(OC)CC1)=O c1(C(N2CCN(C(c3ccnnc3O)=O)CC2)C#N)ccccc1F C1(N(C(CCCc2ccc(C)s2)=O)C)CCCN(C(c2c[nH]cc2C(C)C)=O)C1 C1(CNC(C(C)OC)=O)CCC(NC(=O)C(C)(C)c2ccccn2)C1 c1(CCC(=O)NCCC(OC)OC)ccccc1[N+](=O)[O-] c1(SCC(=O)NC2CN(C(COc3ccc(OC)cc3)=O)C2)cc(C)ccc1C C1(C(=O)NCCC(C)NC(c2ccc(CO)o2)=O)(C(F)F)CCCO1 C1(CC)CN(C(=O)CC2(OC)CN(C(=O)C(C)(C)n3cncn3)C2)CCO1 c1(NC(c2cn(CC=C)nc2)=O)cc(OC)cc(Br)c1.C12CCCC1CNC2=O CC1(C)CC(CNC(c2cccnc2C2CC2)=O)CN1C(=O)Cn1nccc1N c1(CN(C(=O)C(O)C2CCC2)CCCNC(C2CC2(Cl)Cl)=O)ccccc1 c1(C(=O)NC(C)CCNC(C2CC2F)=O)cc(F)cc(S(N)(=O)=O)c1 C1(C(C)(C)NC(C2CCC3CC23)=O)CCN(c2nccc(C(C)(C)C)n2)CC1 c1(CC)sc(C(N2CCC(C(C)NC(=O)CS(=O)CC)CC2)=O)cc1C N1(C(c2cccc(CC=C)c2)=O)CCC(C=CC(=O)NC(C2CCOC2)C)CC1 c1(C(=O)NCC2(NC(c3ncc(Cl)s3)=O)CCOC2)ccc(O)cc1 N1(C(CC(C)CC(C)(C)C)=O)CCC2(CCCC2NC(=O)C2=CCOCC2)CC1 c1(C(=O)NCC(=C)CNC(=O)CCc2ccccc2)ccccc1C(=O)N(C)C N1(C(c2n(CC)ncc2Cl)=O)CC2CCC1C(CNC(c1cc(C#N)c[nH]1)=O)C2 C1(C(N(CC#C)CCOC)=O)CN(C(=O)C(=O)NCC(F)F)CC12CCC2 c1(C(N2C(C)CC(CNC(CC(=C)Br)=O)C2)=O)ccc(Cl)cc1F C(=O)(C(CC(C)CC)NC(=O)Cc1cnn(CC)c1)NC(CCC)C1CC1 N1(C(C(n2ccc(C)n2)(C)C)=O)CCC(NC(=O)C(F)(F)F)C2(CCC2)C1 N1(C(c2ccn(Cc3snc(C)n3)c2)=O)CCCCCC1CCO.N12CC(C1)C2 c1(C(=O)NC(CNC(C=C(CCC)C)=O)CC)ccc(=O)n(CC(C)O)c1 N(C(=NCC(C)C)NCC1CCCCC12CC2)CC(C)(C)SC c1(C(=O)NCCC(C)(C)NC(C(C)Nc2scc(C)n2)=O)ccc(C2CC2)nc1 Cc1cc(C)c(NC(C2CCN(Cc3cc(F)cc(I)c3)CC2)=O)cc1C N1(c2ncc(OC)cn2)CCC=C(C(=O)NCc2nccnc2Cl)C1 C12(C(=O)OCC)CC(CO1)N(C(=O)CNc1ncccn1)C2.C12(CC1)C(=O)N2.SCC C(C(=O)Nc1c(C)c[nH]c1C(C)C)(C(C)(C)C)n1cc(CC(CC)OCC)nn1.OC c1(OC)ccc(C(N2CCCC(NC(C3CC(=C(F)F)C3)=O)C2)=O)cc1Cl C1(NC(Cn2cc[n+](C)c2)=O)CC(CNC(=O)CCOCC(F)F)C12CCC2 n12nc(C3CC3)cc1N1CC(C1)C2=O.C(=O)(C(C)(C)C)OC.CC N1(C(C=C(CC)C)=O)CCC(C2(NC(=O)CN3CCS(=O)CC3)CC2)C1 N1(C(Cc2c(C)noc2)=O)CCN(C(c2cnc(S)n2C)=O)CC1CF c1(C(N(c2nc(C)c(Br)cn2)C2CCCCNC2)=O)ccc2ncccc2c1 c1(CNC(CN(CC(C)C)Cc2cnn(-c3ccccc3)c2)=O)ccncc1 C(CC(C)(C)C(=O)N(CC(C)O)CCNC(C1CCN(C)CC1)=O)SC C(=O)(C(O)(C(F)(F)F)C1CC1)N1CC(O)CC(NC(c2cc(C)c(F)cn2)=O)C1 C(=O)(C1=C(C)CCOC1)N1CCOCC(C(=O)NC(COC)C(N)=O)C1 N1(Cc2ccc(COCC)o2)CCC(C(=O)Nc2cc(Cl)c(C)cn2)C(OC)C1 C1(CC)COCCN(C(C2CCC(NC(c3cncc(O)c3)=O)CC2)=O)C1 N1(C(C2(C)CC(C)C2)=O)CCCC1(C)C(=O)NCCOCCN(C)C N1(C(c2c(C)n(C(C)C)nc2)=O)CCCN(C(C2CC(C)N(C)C2)=O)C(C)C1 c1(NC(c2c(OCC)cccc2)CC)ncnc(N2CCC3(CC2)CC3)c1C C=CCC(C)(CC)C(=O)N1CCC(NC(=O)C(F)C2CCCC2)C(O)C1 N1(CC)CCC(NC(=O)C(CCOCC)NC(c2csnc2Cl)=O)CC1 C#CCC(CC#C)C(=O)N1CCC(CF)(NC(=O)Cn2nnnc2C(C)C)C1 C1(CC=C)(NC(=O)C(F)OC(F)(F)F)CCN(C(c2cc(C)c[nH]2)=O)C1 C(=O)(CC(C)(C)CC(F)(F)F)NCC1CC(NC(C2CC(CC)OCC2)=O)C1 C(C(=O)N(C1CCN(C(c2ccc(C3CC3)s2)=O)CC1)C)(C(C)C)N.C(N)(=O)OC C(=O)(C(F)CCC(C)(C)C)NCC(C)N(C(c1ccc(C)c(O)n1)=O)C N1(C(C2(C)CC=C(C)CC2)=O)CC(C2CCCCN(C(c3cnc(O)s3)=O)C2)C1 c1(C(=O)NCC#CCNC(C=CC)=O)ccc2cc(C(C)C)ccc2c1 c1(C(N2CCC(NC(CCC(=O)NC)=O)CC2C)=O)cnn2c(C)c(C)ccc12 S(=O)(=O)(CCS(=O)(=O)C(F)(F)F)N1C(CC)(OC)CNCC1 C(CCC)(C(=O)N1CC2CC1C2NC(C12CC(F)(C1)C2)=O)=CCC n1(CC)nc(C2CC2)cc1C(=O)NC1CC(NC(=O)CC2(C)OCCO2)C1(C)C C1(C(N2CCC(C(C)NC(c3c(C)scc3)=O)CC2)=O)CSc2ccccc2O1 N1(C(C=CC(=O)OCC)=O)CC2OCCN(C(=O)CN(C)C(C)=O)C2C1 C(C(=O)N1CCCO1)NC(C(C1CC(C#N)C1)NC(C1OC2CCC1C2)=O)=O C1(CC(=O)NCCCNC(C2CCC3(CCC3)OC2)=O)Cc2cccc(Cl)c2O1 O=S(=O)(c1ccc2nc(O)oc2c1)N1CCOCC1CN1CCCC(O)C1 c1(C(N(CC(O)CNC(=O)CCn2ccnn2)C)=O)ccc(CC2CC2)s1 C12(C(N3CC(CNC(C4CCC(O)C4)=O)C3)=O)CCN(C1)S(=O)(=O)C2 C(=O)(CC(F)(F)C(F)F)N(C1CN(C(C(C)C2CC2)=O)C1)C C1(C(=O)NCCC(CNC(COC)=O)O)CCc2nc(C)cn2C1 CC1CN(C(=O)CCCS(N)(=O)=O)CC(C)N(C(=O)Cn2cnc(=N)[nH]2)C1 O=C(C(F)CC1CN(C(C2(Cl)CC2)=O)C1)Nc1cnn(CC2CC2)c1 C(=O)(CCCC(=O)N(C1CN(C(C2CNC(=O)C2)=O)C1)CC)N(CC)CC c1(C(=O)NCC(CNC(c2cc(Cl)cc(C)c2N)=O)C)cnn2c(C)ccnc12 c1(C(=O)NC2C(NC(C3(NC(N)=O)CCCC3)=O)CCC2)cnc2occc2c1 C(=O)(CC(C)CC(F)(F)F)N(CC(C)NC(Cc1nnc(C)o1)=O)C c1(CNC(C)(CCBr)c2nnnn2C2CCC2)cccc2ccsc12 C1(C(N(CCN(C(c2n(CC(C)C)ncc2)=O)C(C)C)C)=O)CC2C=CC1CC2 C(CC(=O)N(C)CC1CCCCCC1)(C(C)(C)C)NC(C(CC)OCC)=O Cc1cnc(N)c(C(N2CC(NC(=O)CCN(S(C)(=O)=O)C)CC(O)C2)=O)c1 c1(C(=O)NCCCNC(C2C3COCC23)=O)cc(Br)c(=O)n(O)c1 c1(NC(C(C)OCCN(C(c2cn(CCC)nc2)=O)C)=O)cccc(Cl)c1C C(C)(C)(CC(F)C(=O)N(C)CC1CC1)NC(C(COCC)C)=O Cc1cc(C(=O)NC2CCN(C(C3CC3F)=O)CC2F)ccc1-c1ccccc1 c1(OCC)ccc(CNC(C2N(C(C3(C(=O)NN(C)C)CC3)=O)CC2)=O)cn1 N1(C(C(C(C)C)O)=O)CCCOC(CNC(=O)CCNC(=O)C=CCl)C1 N1(C(COC(C2C(C)C3C2CCC3)=O)=O)CCOc2ccccc21 C1(C(=O)NC2(CNC(CC(C)n3cccc3)=O)CC2)COC2(CCC2)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C(N2CC3CCC2CC3)=O)CC1)OC c1(C(N2C(CCCC)C(=O)NCC2)C(=O)NCC)cc([N+](=O)[O-])ccc1F O=C(NNc1c(F)ccc(F)c1Cl)c1cccc(S(=O)(=O)N2CCCC2)c1 C1(CNC(CS(=O)(=O)NC)=O)CN(C)CCN1C(=O)Cc1cccn1C c1(C(N2C(C)CN(C(C3CCCC34CCC4)=O)CC2)=O)coc2c1C(O)CCC2 CC(C)C(CCO)NC(=O)CC1(N(C)C(c2ccc[nH]2)=O)CC1 Cc1ccc2nc(NC(c3cc(O)nc(C(F)(F)F)n3)=O)sc2n1 C1(CC=C)CCCCN1C(=O)CCC1CCCN(C(=O)CCC=CC(C)C)C1 Fc1ccc(I)cc1CNCC1CCN(c2ccc(Br)cc2)C1 c1(C(N2CCN(C(Cc3nc(=N)[nH][nH]3)=O)CC(O)C2)=O)coc2c(F)cccc12 C(=O)(CN=S(C)(C)=O)NCCN(CCCN(C)C)C(c1c(SCC)cccc1)=O C1(CC)CCC(C(=O)NC2(CCNC(C3CCC(C)(C)O3)=O)CCC2)CC1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(NC(=O)C(CC)SC)C(C)C1 N1(C(c2cc(C(C)C)cc(C(F)(F)F)c2)=O)C2CCC1C(O)CCC2O C=CCC(N=c1cccc(S(=O)(=O)NCc2cc(C)c(C)s2)[nH]1)c1ccccc1 C1(CCC)CN(C(c2sc(O)nc2C)=O)CCN1C(c1cc(Cl)cs1)=O C(CCCC(=O)NCC(O)CNC(c1cccnc1OCC(F)F)=O)SC N1(C(C(COC)C)=O)CC2CC(NC(c3c(OC)cccc3OC)=O)C(C2)C1 CCC(CC(=O)NC(C)C(C)NC(c1coc(C2CC2)n1)=O)CC(C)C c1(C(=O)NC2CCCC(NC(c3ccc(C)cc3)=O)CC2)ccc2occc2n1 C(c1ccc(C(F)F)o1)=CC(=O)N(C)CC1CCN(C(C(C)OCCOC)=O)C1 c1(OC)ccc(C(CC)NC(=O)Nc2nc(CC(C)C)cs2)c(Br)c1 c1(C(c2nnnn2C(C)(C)C)NCCC2CCN(C)C2)cccc2c1CCCC2 c1(NC(C2C(C)C2C)=O)ccccc1C(=O)OCc1ccccc1 c1(NCC2(NC(C(CC)OC)=O)CCCC2)nccc(COC)n1 N1(C(C2C(CC)OCC2)=O)C2CCCC1CN(C(=O)C1=CC3CCC(C1)C3)C2 N1(C(c2c(OC)ccnc2)=O)CC2(CCC(CNC(=O)CN3CCSCC3)O2)C1 CCCCC(C(=O)N1CCN(C(=O)CONC(=O)OC)CC1)Nc1nnnn1C c1(CC(=O)NC(CO)CCCCNC(c2csnn2)=O)ccc2nonc2c1 c1(CC(N2CCCC(NC(C3(C=C)CC3)=O)C2)=O)ccc(C)c([N+](=O)[O-])c1 C(=O)(CCS(C)=O)N(CC1(NC(CCc2onc(CC)n2)=O)CCC1)C1CC1 c1(C(=O)O)cccc2nc(O)oc12.C(=O)(CSCC(=O)OC(C)(C)C)NCCN(C)CC C(=O)(CC(O)CC(C)(C)C)N1CCC(NC(CCCC#CC)=O)C(C)C1 c1(CCN(C(C2CN(C)C(=O)C2)=O)CCO)n[nH]c2c1CCC2 c1(SC)ccc(C2CC2)cc1.C1(c2cn(C34CN(C3)C4=O)nn2)CCSC(C)C1 C(=O)(CCCS(N)(=O)=O)N1C(CCNC(c2c(C)n(CCO)nc2)=O)CCC1 C1(OC)CC(CNC(c2cnn(C)c2SC)=O)N(C(=O)C=CCO)C1 c1(C(=O)OC)ccncc1C(=O)NCCCCCCN(C(=O)CC1(C)CCC1)C c1(CC(=O)NC(COC)C)ccccc1NC(=O)NC1COCC1OC Cc1[nH]nc2c(C(=O)NCCC3CN(C(=O)CC(C)(C)O)CC(C)O3)cccc12 c1(N(C2CCCN2C=O)C2CCN(C(C(CC)C)=O)C2)cnc([N+](=O)[O-])n1C C(=O)(CCCCC1CC1)N(C1CCN(C(C2CC23CC3(F)F)=O)C1)CCC CCC(CC(=O)NCC(O)CN(C(=O)COc1ccn(C)n1)C)C1CC1 C=CC(C)(O)C(=O)NCC1CCCN1C(=O)CS(=O)CC C(=O)(CCCC(=O)N1CC2(NC(c3cc(OC)ccn3)=O)CC1C2)OCC c1(N2CCC(CC(CNC(=O)OC(C)(C)C)OC)CC2)cc(O)nc(C)n1 n1(CC(=O)NCC2(NC(CC3C(C)OCC3)=O)CCCC2)ncccc1=O N1(C(c2ncc(CC)s2)C(=O)NCCC2(C)CC2)CCCC(CC(=O)OC)C1 C1(C(=O)NCC(=O)OC)CN(C(=O)C(c2cnn(C)c2)O)CC1OC c1(NC(=O)OCCN(C)C)cc2c(cc1OCC(F)C1CC1)OCO2 c1(CN(C)C(c2c(Cl)cnn2C)=O)ccc(CNC(=O)CC2CCC3CC23)cc1 C(=O)(C(CC)CC(C)C)NC(CC#CC)C(=O)NCc1ccco1 c1(C(c2n(CC)nnn2)NCC2CCOC2)cc2ccccn2n1 N1(C(c2cc(Cl)cc(Br)c2F)C(=O)NCCCC)CC2CC(O)C(O)CC2C1 C#CC1(C(=O)NCC2(C)CCN(C(=O)CCc3cnccn3)C2)CCOCC1 C(CNC(c1cn[nH]c1)=O)(CO)NC(=O)COCC1CCCO1 N1(C(C2OCC(C)C2)=O)CCC(CCN(C(=O)CC2OCCO2)C)CC1 N1(C(CC(CNC(CSCCOC)=O)C2CCC2)=O)CCN(C(C)=O)C(C)C1 C(=O)(C(C)C(O)CC(C)C)NCC(C(=O)NC(CCCC=C)C1CC1)OC CC1CN(C(=O)CC2CCC2)CCC1CNC(=O)CCNc1ccccc1Cl c1(C(N2C3CC(NC(c4cn(CC)nc4)=O)(C3)C2)=O)c(Cl)c(CC)nn1C c1(C(=O)NC2CCCN(C(c3ccc[nH]3)=O)C2)cnc(=NCCF)[nH]c1 c1(OC)cc(CN2CCC(O)C(C(=O)NCCCS(C)(=O)=O)C2)ccc1I c1(C(=O)NCC(C)NC(C(C(C)C)N2CCCCC2)=O)cc(F)c(F)c(Cl)c1F CC(C)(O)C(C(=O)NC1CCCC1C(C)(C)C)NC(=O)C(=O)NCC(F)F c1(CN)cn(C)nc1C.N1(C(C(C)SCCCC)=O)CC2(C1)C(=O)N(C)C2 C(CCCCC(=O)NC1CC(NC(=O)C(C)Oc2ccccc2)C1)OC CCCCC(C(=O)NC1CCCC1CNC(c1nccn1C(C)C)=O)N(C)C c1(CC(=O)NC2CCC2CNC(=O)Cc2ccc(Cl)s2)csc(Cl)n1 c1(C(=O)NCC2N(C(C(C3CCCC3)OC)=O)CC2)ccccc1C1(C#N)CC1 N1(C(C(C)CF)=O)CCC2(CCCC(OCC)O2)CC1.C1(C)(C)C(=O)O1.C(=O)CO C1(C(N2CCC(C(C)(C)C(=O)N3CCC(C(N)=O)C3)C2)=O)CC2(CC2)CO1 n1(CC)nc(C2CC2)cc1C(=O)NC1CC(NC(=O)C(C)SC(C)C)C1 C(=O)(C(C)CC(N)=O)NCc1cc(C(=O)NCC2ON=C(C)C2)n[nH]1 CC(CC(=O)NCC1CC1)N(C)C.C1CCCCNC(=O)C(=O)N1 c1(C(=O)NC2CC(NC(c3ccc(C)c(C#N)c3)=O)C2)ccc(S(N)(=O)=O)cc1 c1(C(=O)NCC#CC(=O)NC(CC(C)C)(C)C)cc2ccccc2[nH]1 N1(CCOC)CCC(CN(c2cscc2C(F)F)C(=O)OC(C)(C)C)C1 C1(C(=O)NC(C)(C)CO)CC12CCN(C(c1cc(C(F)(F)F)ccc1F)=O)CC2 c1(C(N2CC(CNC(c3n[nH]cc3F)=O)OCC2)=O)noc2c1COCC2 N1(C(c2ccc(SCC)cc2)=O)CCC(C)(NC(c2ccc(Cl)o2)=O)CC1 C12(NC(=O)CCc3ccc(F)nc3)CCN(C(=O)CC3OCCO3)CCC1C2 C(C(CCC)C(=O)Nc1cccnc1)OC(c1cccn(CC#C)c1=O)=O c1(SC)ccc(C(=O)OC(C)(C)C)o1.C12(Cl)CC1N2C(=O)NCCc1nncs1 N1(C(C(C)NC(C=C)=O)=O)CC2OCC(C(=O)NC)C2C1 Cc1cnc(C(N2CCN(C(c3nccc(Cl)c3F)=O)CC2C)=O)c(F)c1 C(=O)(CS(=O)(=O)C1CC1)NC1CC(CNC(C2(C#C)CCC2)=O)CC1O c1(NCn2ncc(C(OC)OC)n2)ncn(C)c(=O)c1Br N1(C(c2n(C(CC)CC)nc(C)c2)=O)CCOC2CCN(C(C3CC3F)=O)CC12 C1(C(C)C)CN(C(c2ccccn2)=O)CCN1C(=O)C=Cc1csc(Br)c1 c1(NCCC(C)NC(c2ccc(Cl)cn2)=O)cc(O)nc(O)n1 C1(C(=O)NCCOCC#C)CCCCCCN1C(c1conc1C(C)C)=O C1(C)(C(=O)NCCC2(C(=O)NC(C=C)C3CC3)CCCC2)CCCCCC1 C1(C(=O)NCC(C)(C)OCC(=O)NCCOCF)CCCC12CCOCC2 N1(C(C(C)Cc2ccco2)=O)CCCC(C2CCN(C(C34CC(F)(C3)C4)=O)C2)C1 c1(C(=O)NCC2CC(NC(=O)OC(C)(C)C)C2)cnccc1Cl c12ccc(cc1F)oc2=O.N1(C(=O)NC)CC2CC(CC34COCC3C4)C2C1 N1(C(N)=O)CCCC(c2nnnn2CCF)(NCc2cc(Cl)cc(Cl)c2)C1 N1(C(CC(C)C)=O)CC(NC(c2nn(C)c(C(F)(F)F)c2Cl)=O)CCC1C Cc1ccc(OC(=O)CCc2cnccn2)cc1C.c12ccc(cc1)c(=O)[nH]2 C1(C(C)(C)O)C(=O)N1.C1(C)(C)C(=O)N1.C1C(C)C1C.CC(C)OC(C)=O c1(C(=O)NCCCCCNC(c2c(OC)scc2)=O)nccc(Cl)c1Cl N1(C(c2ccc(OC)nn2)=O)CC(NC(c2nc(C)nn2C)=O)CC1(C)C c1(C(C)C(=O)N2CC(CCNC(=O)CCSc3ccccn3)C2)cncnc1 c1(C(=O)NCC2N(C(C(C)c3ccsn3)=O)CCOC2)c(N)nn2ccccc12 n1(CCC(=O)NCCN(C(c2ccsc2Cl)=O)C2CC2)ccccc1=O C1(CNC(CN(C)C(c2ccsc2)=O)=O)CN(C(C2(Cl)CC2(F)F)=O)CCO1 n1(CC)cc(NC(=O)C(CC(F)F)NC(=O)Cc2ccc(O)cn2)ccc1=O c1(SCC(=O)N(CC(C)NC(C2(C(F)F)CC2)=O)CC)nnnn1C1CC1 C(=O)(C(O)Cc1cn(C)cn1)NC(CNC(C1(C(=O)NC)CC1)=O)C c1(SC)cnn(C)c1C(=O)NCC12CC1CN(C(=O)C(C)C1(O)CCC1)C2 S(=O)(=O)(c1ccc(NC2CCOC(C(=O)O)C2)cc1Cl)N(C(N(C)C)=O)CCO C1(CC(=O)NCCC2CN(C(C)=O)CCO2)(CNC(C)=O)CCCCC1 N1(C(c2ccc(C(C)(C)C)o2)=O)CC(F)(F)CC1CNC(C1CCC=CO1)=O N1(Cc2cccc(C(C)C(F)(F)F)c2)CCC(O)C(C(=O)Nc2cn(C)cn2)C1 c1(NC(CC2OCCN(Cc3c(C(C)C)cccc3)C2)=O)cccn2ncnc12 c1(C(=O)OC)cccc2nncn12.C#CC1CCC(C(N2CCN(CC)CC2)=O)CC1 C(=O)(C(O)CC(C)(C)C)N1CC(CCNC(c2c(C)sc(O)n2)=O)OCCC1 C1(CC(=O)N(C(C)CNC(=O)CN(C)CCO)C)(C(=O)OC)CCCO1 N1(C(C(COC)O)=O)CCC2(NC(c3cncc(CO)c3)=O)CCCCC12 CC(C)(C)C(CC(=O)NC1C2CN(c3ncnc(Cl)c3Br)CC12)C(F)F CC(CCC(=O)NCCN(C(c1cccc(-c2cnn(C)c2)c1)=O)C1CC1)N(C)C c1(CC(N2C(C)(CC(=O)NCCCNC(C)=O)CC2)=O)ncc(F)cc1F C(CCCCC(=O)NCC1CCC2(CCC2)O1)NC(C(CCC)C)=O N1(C(CONC(C(OC)OC)=O)=O)CCC2(CCOC2)C1 C(=O)(C1=CC(C)(C)C1)N1CCC(C(C)NC(C2(c3ncco3)CCC2)=O)C1 c1(OC)ccc2c(C(N3CC4(CNC(C5(Cl)CC5)=O)CCC3CC4)=O)cnn2c1 c1(CSC(C)C(=O)NC2CC=CCO2)cn(CC2CNC(=O)O2)nn1 CCCCCCOCC(=O)N(CC(C)NC(=O)CC(C)c1ccncc1)CC c1(CC)cc(Cl)ccc1C(=O)NC(C)C(C)NC(=O)C(C)(C)NS(C)(=O)=O c1(C(=O)NCCN(C(C)C)C(c2cncc(C(N)=O)c2)=O)ccc(=O)oc1 N=c1nc2c(c[nH]1)CC(C(=O)NC1(CNC(c3cc4c([nH]3)CCCC4)=O)CC1)CC2 C12(C(N(C3CN(C(=O)CC4CCCCO4)CC3O)C)=O)CCC(F)(CC1)C2 O=[N+]([O-])c1cc(F)c(CN(CCCOCC2CCOC2)C)c(F)c1 Cn1nc(C(N2CC3CC2(CNC(C2CC(O)C2)=O)C3)=O)cc1C#N N=c1[nH]cnc2cc(C(N3C4CCC3C(CNC(c3ccc[nH]3)=O)C4)=O)ccc12 C1(NC(C2C3C(NC(C(C)=C4CC4)=O)C4C(C3)C42)=O)CC(C)(C)C12CCC2 Cc1cc(=NC(=O)C2CCOC2NC(=O)N2OC3CCC2CC3)[nH]n1C C1(N(C)CCNC(c2cc(Br)sn2)=O)CCCN(C(=O)N(C)C)C1 C=CC(C(F)(F)F)NC(=O)C(CCC1CCC1)NC(=O)CCCn1ccnc1 CC(=O)CCCC(=O)N1CCN(c2cc(C(C)(C)C)ncn2)C(CO)C1 c1(C(N(CC(CC)NC(c2ccc(C(N)=O)o2)=O)C)=O)ccc2occc2c1 O=S(=O)(c1ccc(NCC2CC3CSCC3C2)c(Cl)c1)NCC(c1ccsc1)O N1(C(C2CCN(CC)C2)=O)CC2(CNC(=O)CO2)C1 S(=O)(=O)(c1cccnc1)NCc1ccc(NC(c2cn(C3CCC3)nn2)=O)cc1 C(=O)(C1=CCCOCC1)NC1C(CC)CN(C(c2occc2Cl)=O)CC1 c1(CN2CC(C)(C)OC(CO)C2)cccc2ncccc12 Cc1nc2ncccn2c1C(=O)Nc1nnc(Cc2ccccc2)s1 C(=O)(C#CC1CCCCC1)N1CC(C)(CNC(C2CSCC(=O)N2)=O)OCC1 C1(CC)C(NC(=O)Cc2ccn(C3CC3)n2)CCCN1C(c1n[nH]cc1Cl)=O C1(NC(c2cc(OC)no2)=O)CC2CC(NC(=O)C=C(C)C(C)(C)C)C2C1 c1(NC(CC2C(NC(C(C)OCCOC)=O)CC2O)=O)cc(C)c(F)cc1O C(=O)(C1CCOc2ccccc21)N1CC(CC=C)(NC(=O)C(C)CC)C1 C(=O)(C1SCc2cccnc21)N1CC(CCNC(CN(CCC)C)=O)C1 C1(CN(C(C(C)O)=O)C)CN(C(c2nn(C(F)F)cc2Cl)=O)CCO1 O=C1CCN(C(C2CC3(CC3)CN2C(=O)CC2CC3CCC2O3)=O)CCN1 CCC(C(=O)NCC1(C(=O)NCC2CC(CO)CO2)CC=CC1)NC(N)=O c1(NC23C(CN(C(=O)OC(C)(C)C)C2)CCCC3)cc2c(nc1O)CCCC2O N1(C(CCN(S(CC)(=O)=O)C)=O)CC(CN(C(=O)C(C)SC)C)C2(CC2)C1 N1(N(C(c2ccc(CCC)s2)=O)CC2(C(N)=O)CC2)CC2CCCC2C1 C1(C)(NCC(C)(F)Cn2cc(C(c3ccc(F)cc3)O)nn2)CCS(=O)(=O)CC1 CC(C)(C)C(CO)C(=O)NC1(CCNC(=O)C(O)C2CC2)CCC1 c1(CN2CC(C(=O)NCCOCC#C)SCC2)cc(F)cc(I)c1 N1(C(c2c(N)c(F)ncc2)=O)CC(NC(c2ccc(CO)o2)=O)CC12CCC2 N1(C(Cc2cn(C)nc2)=O)C2CCC(C2)C1CNC(c1cc(F)c[nH]1)=O N1(C(CC2CCCC(C)(C)C2)=O)CCC2(CC1)CC2CNC(=O)CSCC(N)=O c1(CC)ccc(O)c(C(N2CCC(CNC(=O)CC(CC)C3CC3)C(O)C2)=O)c1 CC1=C(C(=O)NCCC(C)N(C(=O)COc2cccc(O)c2)C)CCCC1 N1(C(C=COC(C)=O)=O)CC(O)(CO)C1.C1(C(=O)N)CC(=C2CCC2)C1 C1(C(=O)NCC(COC)C(C)C)CN(C(C2CC3(C2)CC(O)C3)=O)CC12CC2 N1(C(C2(C=C)CC2)=O)CCCCC1C1(NC(c2ncnn2CC)=O)CC1 Cc1cc2cc(-c3cn(C4CC(NC(C5CCCC5(F)F)=O)C4)nn3)cnc2[nH]1 C1(F)(CNC(CSC(C)C)=O)CCN(C(c2sccc2Cl)=O)CC1 CN1CC(C)(C)CC1C(=O)NC1CC12CC(NC(=O)CC1(C)OCCO1)C2 C1(C(=O)NC2C=CCN(C(=O)C=CC3CCCC3)C2)Cc2ccccc2S1 N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(c2cc(C)c(C)[nH]2)=O)C1 C=CCCC(C(=O)N1CCC(C)(C#N)C1)NC(c1nnn(CC)c1C)=O c1(C(N2C3C(NC(c4coc(CO)c4)=O)C(CC3)C2)=O)ccnc2ccccc12 C1(O)(CNC(C(C)CC2CCC2)=O)CCN(C(C2CCC(O)CN2C)=O)CC1 CC1(C)CCOC(C(N2CC(O)(C(F)C(=O)NC3CCC4CC3CO4)C2)=O)C1 C(CCCC(=O)N1CCCCC1c1ncc[nH]1)n1cc(-c2c(C)occ2)nn1 N1(SCCCNC(=O)C(O)C2CCCC2)C(=O)CCC1C(=O)N(C)CCOCC C(CCC(O)C(=O)NCCOC1CCCC1)NC(c1nn(C)c(CO)c1)=O Cc1cc(NC(=O)CN2CCC(NC(=O)CCc3ccoc3)C(O)C2)ccc1F C(=O)(CCCCN=[N+]=[N-])NCc1nc(C)c(C(=O)NCCN2CCCCCC2)o1 C1(C(N(CCOCCC(=O)NCC(C(C)C)C)C)=O)CC(=O)OC1(C)C c1(C(=O)NCCCCC2CN(C(C(COC)C)=O)C2)coc2c1CS(=O)(=O)C2 CC1CN(C(C2CN(C)C2)=O)CC1NC(C1CCCN1C)=O c1(CC)nc2n(n1)CCCC2NC(=O)C(n1cc(-c2ncc(C(=O)O)o2)nn1)C c1(C(N2CC(O)(CCNC(c3c(C)cn(C)c3)=O)C2)=O)c[nH]c2cccc(F)c12 C1(NC(c2ccc(C)nn2)=O)CCN(C(=O)Cn2nccn2)CC1CO c1(OC)ccc(C(=O)NC2CC(CNC(C3CCC(C#N)C3)=O)C2)c(Cl)n1 c1(C(=O)NCC2CC(C)N(C(C3C4CCCC34)=O)CC2)ccc(F)c(F)c1F C1(O)(C(C)NC(CC2(OCC)CCCC2)=O)CCN(C(C2CCSCC2)=O)CC1 C1(CC)(C)CCCN1C(=O)CC1(N(C(=O)CC2(C)CCC2)C)CC1.OC CN1CCN(CC(=O)N(C23CC(NC(=O)CC4CC5COCC45)(C2)C3)C2CC2)CC1 C1(NC(c2sccc2CC#N)=O)CCN(C(C23CCC(C2)C3)=O)CC1O C1(N(C)C(c2ncoc2-c2cccs2)=O)CN(C(C2(Cl)CC2)=O)CC1(C)C C1(CCNC(C(C)(C)C2CCC2)=O)CCCCN1C(c1cn(C(F)F)cn1)=O c1(N2CCC(C)(NC(C3OCC3(C)C)=O)C2)ccc([N+](=O)[O-])cc1C(F)(F)F c1(NC(=O)NC(CC)Cc2ncc(-c3ccc(Cl)cc3)s2)cccc2cccnc12 N1(C(CCCCC=CC)=O)CCCC(C)(C)C1CNC(=O)Cn1nccc1C S(=O)(=O)(c1cnc(NCCC(O)C2CC2)c(Cl)c1)NC1CCC(CCCC)CC1 N1(C(C(C=C)O)=O)CC2(COC(CNC(=O)CCCn3nc(C)cc3C)C2)C1 c1(C(N(CC(C)CNC(c2nc(C(C)(C)C)no2)=O)C)=O)ccc(C2CC2)cc1 c1(C(=O)NC2C(C)(C)CN(C(=O)CC3CCOC3)C2)ccc2ncccn12 c1(C(N2C(C(N(CC)CC3CCCC3O)=O)CCCC2)=O)ccc(C2CC2)nc1 C1(NC(C(C)C2CC2)=O)CCC2(CCN(C(=O)C(C)(C)C3CCC3)C2)C1 C1(CC(=O)NCCN(C)C(c2sc(C(C)(C)C)nc2C)=O)CC2C=CC1C2 C1(CC)(NC(=O)C(C)SC)CCCN(C(C2(c3ccc(F)cc3)CC2)=O)C1 c1(CCC(=O)NC(C)CN(C)C(C23CC(C)C2C3)=O)c(Cl)cncc1Cl C(CCCCC(=O)N1C2CCC1CNC2)n1cc(-c2c(C)cccc2)nn1 N1(C(CCCOCC)=O)CCC(C2CCCN(C(c3ccncn3)=O)C2)C1 C(=O)(CCCC(=O)c1ccccc1)NC(C1CN(C(=O)CC2CSC2)CCO1)C Cc1[nH]c(=NCc2cnc(O)nc2O)sc1C(=O)Nc1ccc2c(c1)CCC2 C(C)(C(=O)N(CCCOCCNC(=O)CCN(C)C(C)C)CC)OCC C1(C(=O)NCCN(CCCc2cc(C)c(F)nc2)C)C2C3CC4C1C1C2CC3C41 C1(=O)CCC(=O)N1Sc1ncoc1CNC1CCCC1.c1(C(C)(C)C)ccsc1 N1(C(Cc2cc(C)no2)=O)CC2=C(C1)CN(C(C1COC3COCC3O1)=O)C2 C(=O)(C1=CCCN(Cc2cc(Br)ccc2C)C1)Nc1cccc(CCC)c1 c1(C(=O)NC2C(C)CN(C(c3ccc(O)cc3)=O)C2)nccc2n[nH]cc12 c1(C(=O)NCC2C(NC(Cc3c(C)n(C)cn3)=O)CC2)cc2c(cc1O)OCO2 C(C)(CCC(=O)NC(C)CCN(C(=O)CCCc1sccc1C)C)OCC Cc1[nH]nc(C(=O)NCCC2(O)CCN(C(c3coc(O)n3)=O)CC2)c1[N+](=O)[O-] C(CC(C)N=c1[nH]c(=NCCc2c(F)cncc2F)c2cccc(F)c2[nH]1)SC C(=O)(CCCCC(F)F)NCCNC(C(c1cn(C)nc1)=O)=O C1(CNC(CC(C)(C)F)=O)CCN(C(=O)C=CC2CCOCC2)CC1(F)F C12(C(=O)NCCC3CCN(C(Cc4cc(OC)no4)=O)C3)CCC(C1)C(C)(C)O2 c1(CC)ccc(C(=O)N(CC(O)CNC(c2cnn(C)c2C(F)F)=O)C)cc1N Cc1ccc(N)c(C(=O)NCC2CCCC(NC(=O)CN=S(C)(C)=O)C2)c1 N1(C(Cc2c(C(C)C)con2)=O)CCOCC1CNC(=O)COCC(F)(F)F c1(OC)cncc(C(N2CCC(C(C)NC(C3(CCF)CCC3)=O)C2)=O)c1C c1(OC)ccc(O)c(C(N2CCCCC(NC(=O)Cc3cnc(C)s3)C2)=O)c1 c1(C(N2CC3C(CNC(=O)CC4CC4(Cl)Cl)C3C2)=O)n[nH]c2c1CCC2 C#CC1(C(N2CCC(N(C(=O)C(C)C3CC3)CC3CC3)CC2)=O)CCCC1 N1(C(c2cccc3c[nH]nc23)=O)CCOC2(C1)CN(C(C13CCCC1CC3)=O)C2 c1(CC(=O)NCC(CO)NC(C(c2c(OC)cccc2)O)=O)cc(F)cc(F)c1 C(=O)(C(O)CCCNC(C1(C(C)(C)O)CC1)=O)NCCn1c(C)ncc1 N1(C(c2scc(COC)c2)=O)CCC(CO)C(NC(c2csc(Cl)c2Cl)=O)C1 CC(C(=O)NCC1CC1CNC(C1CC2(CCC2)CO1)=O)S(C)(=O)=O CCCCCCC(CC)C(=O)N1CCC(C2CN(C(=O)CCCC(C)C)C2)CC1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC(C)(C)NC(=O)CC1OCCO1 CCC(CC)CC(=O)N1CCCC(C2CCCCN2C(=O)C(C)=CC(C)(C)C)C1 C1(NC(c2cnc(C3CC3)s2)=O)C2CCC1CN(C(Cn1ncc(C)c1)=O)C2 C(=O)(CC(C(F)(F)F)NC(c1nnn(CC)c1C)=O)NCCCC=CC C#Cc1ccc(C(=O)N(CCN(C(=O)C=CSC)C)C(C)C)cc1F c1(NC(CCN(C(=O)CC2CCCOCC2)CC)=O)ccccc1F C1(C(=O)NC(CNC(c2ccc(C(C)C)s2)=O)C(C)C)OC2CCC1CC2 C12(C3CCN(CC3)C1=O)CCC2.CS(=O)(=O)CCc1cn(CC2CCC2)nn1 C1(C(=O)NC(C)(C)CCNC(C2CC(O)C2)=O)COCC1(C)C C1(Nc2cccc(OC)c2)CCN(C(=O)C(N2CCCC(O)C2C)=O)CC1C c1(OCC)ccsc1C(N1CC=CC1CNC(c1cc(OC)ns1)=O)=O C=CCC(CC)C(=O)NC1(C2CN(C(=O)C(=Cc3cnn(C)c3)C)C2)CC1 CCCCC(C)C(=O)NCCOCCNC(C1(c2ccccc2)CC12CCC2)=O N1(C(C(=O)N(C)CCOc2ccccc2)=O)C2CC2C2CC12 C1(CNC(CC=CCC)=O)CC2(CCN(C(=O)CCSC)C2)CO1 CCC(C)C(C(=O)NC1CCCC1NC(c1cnc(C(F)F)s1)=O)OC C1(C)(CC)CC(NC(c2ccc(C)o2)=O)CN1C(=O)Cc1ccc(C)nc1 N1(C(C(c2cccnc2)NC(C2C(C)=CCS2)=O)=O)CCn2c(C)cnc2C1 CCC(C(=O)NCCC1(NC(c2cc(C3CC3)ccn2)=O)CCC1)C(C)(F)F N1(C(C2CC3(CN(C(C4CC=CC4)=O)C3)OC2)=O)CCc2cnccc2C1 Cc1nc(C)c(C(N2CCC3CN(C(C4(C(=O)N(C)C)CC4)=O)CC23)=O)c(C)n1 c1(C(=O)NCC(C(C)C)NC(C2CC=CCO2)=O)nn2ccccc2c1Br N1(C(c2nncc(CCC)c2)=O)CCC=C(CNC(=O)CCCC(C)C)C1 N1(C(C(CCC)(C)C)=O)CC=C(CCNC(C2CCC23CCCO3)=O)CC1 C=C(C)C1OCCC1C(=O)NC1CC(CO)N(C(C2CN(C(C)=O)C2)=O)C1 c1(-c2cnc(OC)s2)nc(C2OCCc3ccccc32)nn1CC(C)C N1(C(c2c(C)nn(C)c2)=O)CC2CCOCC2(NC(=O)Cc2ncc(Cl)s2)C1 c1(C(N(C)CC2(NC(C3CCC3(F)F)=O)CC2)=O)nc(-c2nc[nH]n2)sc1C1CC1 c1(CCC)ncc(C(=O)NCCCOC)s1.c1(C(=O)NCCCC)cnc(Cl)[nH]1 C1(C(=O)NCCC(=C)CNC(c2cncc(Cl)c2C)=O)C2CCCCCC12 CC1CCCN(C(n2cc(CCC3CC4CCC3C4)nn2)C(=O)NCCCF)C1 c1(C(=O)OC)ccc(C(=O)NCC(C2CCCC2)NC(c2cncn2CC)=O)s1 N1(C(C(C)=C(CC)C)=O)CC2(CCCN2C(c2cccc3scnc23)=O)C1 c1(C(C(=O)NC2(CC)CCC2)F)ccc(F)cc1.C12CCN(C1)C(=O)C2 c1(CCC)ccc(C(N2CC(Oc3ccc(O)cc3)C2)=O)cc1[N+](=O)[O-] C1(NC(c2c(OCC=C)cccc2)=O)CCCC2CN(C(=O)CC3(C)CC3)CC12 C1(CCOC)(NC(c2ccc(CO)[nH]2)=O)CCN(C(=O)CCC2CCCC2)CC1 C1(NCCC(=O)NCCOCCCN(C(c2c(C)snc2)=O)C)CCCC1(F)F C1(CC(=O)N(C(C)C)c2ccsc2)C2CN(C(c3csc(C#N)c3)=O)CC12 N#Cc1cc([N+](=O)[O-])cnc1NC(C1CCCC(Nc2nccc(CO)n2)C1)=O C#CCCCCCC(=O)NC(C)CC(C)NC(=O)C(C)NS(=O)(=O)CCCC C1(NC(C(OC)OC)=O)C2CC(O)C1N(C(c1cccc3nn[nH]c13)=O)C2 Cc1cc(=NC2CC(C)NC(C)C2)[nH]c(=NCCCOC2CCS(=O)(=O)C2)[nH]1 C(=O)(C(C)C(=O)N1CCCCC1C1CCN(C(=O)CCc2cnn(C)n2)C1)OC N1(C(C2(COC)CCCC2)=O)CCCC(O)(CNC(c2sccc2C2CC2)=O)C1 C(=O)(CCCC(F)(F)CO)NCCCCCNC(CC1C(C)(C)CCCO1)=O C1(NC(c2c(CNC(=O)CSc3cn[nH]c3)cco2)=O)CC2(CCC2)C1 CCC(CCC(=O)N1CC(C(N)=O)(CNC(c2cc(SC(C)=O)oc2C)=O)C1)OC c1(OCC(N2CC(O)(CNC(C=CCCC)=O)C2)=O)c(Cl)cc(C)nc1CC C(=O)(C1=NOC(C)C1)NC1C(CNC(C2C(CC)C2)=O)CCCC1.c12cc-1on2 c1(Sc2ccc(NC(C34CCC(CC3)C4)=O)cc2)c([N+](=O)[O-])ccc(Cl)c1Cl CC(C)C(C(=O)N1CC(O)C(O)C1)n1cccc1.C12(CC1)C(=O)NC2 N1(C(C(CN(C)C)O)=O)CCC(CNC(=O)CCc2ccc(F)cc2F)C1(C)C CCCC(CC)(c1nnnn1Cc1ccccc1)NC1(C)CC2CCC1O2 S(=O)(=O)(c1ccc(Br)cc1Br)NCC1OCCN(C(C(CCCC)O)=O)C1 N1(C(c2c(CC)nn(C)c2)=O)CCCC(CNC(c2ccnc(F)c2F)=O)CC1 C1(C(N(CC(C)NC(c2ccnn2CC#N)=O)C)=O)CCC(=O)C1 C1(COC(c2csc(COc3ccccc3)n2)=O)CC(O)C12CCC2 N1(C(CCc2cn(C)nc2)=O)CC(C(F)(F)F)CC1CNC(C1C(C#N)C1(C)C)=O c1(CN=C(NC2CCN(C(C(C)C)=O)C2)NC2CC2)cccc2[nH]ccc12 C(=O)(C(C)(O)CCc1ccccc1)NC1CC(NC(C=C(CC)CC)=O)C1 c1(-c2cn(CCC(N3CC(C(=O)OC)C(=O)CC3)=O)nn2)cccc(O)c1F C(CCS(=O)(=O)c1cccc(Br)c1)c1ccc2onc(C)c2c1 c1(OC)ncc(C(N2CCN(C(=O)C(CC(C)C)N(C)C)C(C)C2)=O)cc1Cl c1(C(c2nnnn2CCC=O)NCC)cnc(OC)cc1C.CCCCCCOCC c1(NCc2ccn(C3CC3)n2)cc(NC2CCC3CC23)ncn1 N1(C(c2ccc(F)cn2)=O)CCC(NC(C2(n3ccnn3)CC2)=O)C(F)C1 Cc1ccc(C(N2CCC(C)C2CNC(C2CC(=C3CC3)C2)=O)=O)cc1CO c1(C(N2CCC(NC(=O)CNc3nccs3)C(F)C2)=O)ccccc1[N+](=O)[O-] N1(C(C2C3(CCN(C(c4ncccn4)=O)C3)C2)=O)CCSC2(CCC2)C1 c1(C(=O)NCC(CNC(c2c(C)cco2)=O)C)cnc(CC(C)C)cn1 CC(C)C(C#N)C(=O)N1CCCC(N(C)C(c2ccc(N(C)C)cn2)=O)CC1 CN=c1[nH]cc(C(=O)NCC2CN(C(C3(O)CC3)=O)CCO2)s1 C(=O)(C(C)(F)C(F)(F)F)NC(CC1CN(C(C2(SC)CCC2)=O)C1)C CC1(C(N2CCC(CCc3cn(-c4cccc(N)c4)nn3)C2)=O)CCNC1=O C(=O)(CS(=O)CCC(F)(F)F)NCCCCn1cc(CCOC(C)=O)nn1 C(c1ccc(Cl)cc1F)=CC(=O)NCC(CNC(C1CC2CC2C1)=O)OC C1(N(C(C(c2ccccc2)C)=O)C)CC2CC1N(C(c1n[nH]cc1Cl)=O)C2 CCC(Cc1ccccc1C)C(=O)N1CCC1CNC(C1(C(=O)NCC=C)CC1)=O.OC c1(OC)ncc[nH]c1=NC(=O)CC(N)C(C)(C)C C#CCC(CC(F)F)NC(c1nc(CNC(c2nnsc2N)=O)oc1C)=O C1(NC(C2OCCC(C)(C)C2)=O)CCC2(CCN(C(C3(CO)CCOC3)=O)C2)C1 CC1(C2(C(=O)NC3CN(C(=O)CN=[N+]=[N-])CC3C(F)F)CC2)CC1 C(C(C)(C)C#CC(=O)NCCC1(C)CCCO1)NC(C(C)(C)OC(C)=O)=O C1(F)(CNC(C=CCOC)=O)CCCN(C(=O)C(C)(C)Oc2ccccc2)C1 C1(NC(CN(C)CCO)=O)CCC2(CC1)CC2NC(c1ccc(C#N)c(F)c1)=O C1(NC(CS(CC)=O)=O)CC2(CCN(C(c3cc4c(cn3)CCCC4)=O)CC2)C1 N1(C(CC(C)(C)O)=O)CC2(C1)CN(C(=O)C1=NOCC1)CCO2 C1(NC(Cn2c(C)ncc2)=O)CN(C(=O)CCN2CCCC2)CC2CC12 c1(SC)cc(C(=O)NC(C)C(C)(C)NC(c2ncn(C)n2)=O)ccc1Br Cc1cc(NC(=O)NC2CCC2)n2nc(C)cc2n1.c12ccc(cn1)NO2 c1(OC)cccc(CNC(=O)CSC)c1.C1(C(N2CC(OC)C2)=O)CCOC(C)C1 N1(C(CCCN(C(=O)OCC)C)=O)CCN(C(=O)C(F)(F)COC)CC(O)C1 CC1(F)CCN(C(=O)C(C2CCCC2)NC(=O)Cc2cccnc2)CC1 Cc1cccc(N(CC(O)C(C)(C)C)CCCO)c1 c1(C2(NC(CCN(c3ccccc3)C)=O)CC2)ccccc1F Cc1cc(=NC(=O)C2C3CC4C(C3NC(=O)CC(O)CN(C)C)C24)[nH]n1C N1(C(C=C(C)C(C)(C)C)=O)Cc2ccccc2C(CNC(=O)OC(C)(C)C)C1 Cc1ccc(CN(C(=O)C(=O)Nc2ccnn2C2CCOC2)C)cc1 N1(C(c2cc(CSCC)on2)=O)C2CCC1CN(C(=O)CC1CC13CC3)CC2 C(CCCCC(=O)N1CC(C(F)(F)F)CC1CNC(=O)C=C(C)C1CC1)OCC Cc1cc(CC(N2CCCCC2CCc2ccccc2)=O)cc(F)c1 N(C)(C1=NS(=O)(=O)c2ccccc21)Cn1c(C)nn(CC(=O)NCC(=C)C)c1=O CCCCCCC(CC)NC(c1cccc(NS(=O)(=O)c2cccs2)c1)=O c1(C(N(CC(=O)NCCOC2CCCCC2)CC)=O)cc(O)nc(O)n1 c1(OCCC(=O)NC2(CF)CCN(C(C(CCC)O)=O)C2)ccc(Cl)c(F)c1 C(=O)(CC1OCc2ncccc21)NCc1scc(CNC(CCC(C)C)=O)n1 n1(CC)ccc(C(=O)N(C(C)CNC(=O)C=C(C)C(C)(C)C)CC)c1C N1(C(Cc2cn(C)nc2)=O)CC2CCCC2(NC(C2Cc3nccn3C2)=O)C1 N1(C(c2cccc(C)c2)=O)CC(CNC(C2C(C)C2C)=O)CC12CCC2 N1(C(C=CCC(C)(C)NC(C2C(OC)(OC)CC2)=O)=O)CCC(C)C(C)C1 C1(CNC(C2(C)N(C)CCC2)=O)CC(C)(C)CN1C(c1ocnc1C1CC1)=O c1(OC(CCC)=O)ccc(CN2CCCN(C(C)C)CC2)cc1 C(=O)(CC(F)(F)C(F)(F)F)NC1C(NC(C2N(CC)CC2)=O)CCOC1 Cc1noc(NC(C2CCCN(S(=O)(=O)Cc3ccc(Br)cc3)C2)=O)c1C C1(CCC(C)C)CCCN1C(=O)C(=O)NCC1CCN(C(=O)NC(C)(C)C)C1 CC(C)C(F)(F)CC(=O)N1CCCC1CNC(=O)CCC(=O)c1ccc(O)cc1 C(=O)(C1COc2ccccc21)NCC1(C(N)=O)CN(C(C=C2CCC(C)C2)=O)C1 C12(C(=O)NCc3cc(COC)on3)CC(CN1C(=O)Cc1cscc1OC)C2 c1(C(=O)NC2CCN(C(C=Cc3occ(C)n3)=O)CC2O)cc2sc(C)cc2s1 CN1CCOC(C(N2CC(C(=O)NCCNC(C3(O)CCN(C)C3)=O)C2)=O)C1 N1(C(CCC=C)=O)CC2(NC(c3cnc(C(C)(C)C)nc3)=O)CCC1C2 CN1CCN(C(c2occ3c2CCC3)=O)C(C(=O)NC2CCCSCC2)C1 C=CCC(CC=C)C(=O)N1CCCC1C(=O)Nc1ccc(F)c(CO)c1 C(CNC(=O)CCc1cnn[nH]1)(CNC(=O)CCOCCN(C)C)OC C1(C(NOCCOC)=O)(CNC(C2COCC2C(=O)OC)=O)CC2(CC2)C1 C1(C(N2CCC(C(C(=O)NC(COC)(C)C3CC3)C)C2)=O)CCCCC1(C)C c1(CCOC(C23C(CN(C(=O)OC(C)(C)C)C2)C3)=O)cccc(C#N)c1 C(=O)(C1=C(Cl)CCOC1)N1CC(CNC(=O)CC(C(F)F)c2ccc(F)cc2)C1 c1(CCCC)cc(C(N2CCCC(NC(=O)CCCNC(C)=O)C2)=O)c(C)o1 N1(C(CCOCC#C)=O)CC(NC(=O)CS(N)(=O)=O)CCC1C C(CNC(C1CC12CCOC2)=O)(CC)(CC)NC(CC1CC(=C)C1)=O C1(C(=O)Nc2nc(C(C)C)no2)(CNCC2(C=C)CCC2)CCCCC1 c1(SC)nc(C(F)(F)F)cc(=NC2CCN(CC3(F)CCOC3)C2)[nH]1 C(=O)(CCCCN=c1nc(N2CCS(=O)C(C)(C)C2)c2c([nH]1)CCS2)NC(C)C C1(NC(C(=O)NC(c2cn(-c3cccnc3)nn2)C)=O)CCC(C)CC1 c1(NC(C2CCCN(C(=O)C(F)(F)F)C2)=O)ccc2c(c1)OCO2 c1(C(=O)NCC23N(C(c4nc(C)sc4)=O)CC(C2)C3)cc2ccc(F)cc2s1 O=C(CCc1nc(C2CCOCC2)no1)NNC(=O)CSc1ccccc1Br c1(Cn2cc(-c3cnn(C(C)C)c3)nn2)nc(C)c(NC(CSCCC=C)=O)o1 N1(C(C(CCSC)O)=O)CCC(N(C(=O)CCc2ccsc2)C)C2(CC2)C1 CCCCCC(O)CC(=O)NC1CC(NC(c2ncccc2OC)=O)C1 O=C1CC(C(=O)NC(C(F)(F)F)C2CC2)c2cccnc2N1 N1(C(C(C)C(C)O)=O)CC2(C1)CN(C(=O)Cc1ccns1)Cc1ccccc1O2 C(CC(C)C)(C(=O)NCc1nc(C(N)=O)co1)NC(C(CCSC)O)=O N1(C(C2(NC(CCC)=O)CCCC2C)=O)CC2(CCC(C)OC2)C1 c1(C(=O)NC2(CF)CN(C(C(c3cnn(C)c3)C)=O)C2)cnc2c(c1)NCC2 N1(Cc2sc(C)c(I)c2)CCC(C(=O)O)C(C(C)C)C1 N1(c2cc(N3CCN(C(CCC)=O)CC3)nc(C)n2)CCC(C2CNC(=O)C2)C1 Cc1ccc(Cl)cc1OCC(=O)N(C1CCN(C(c2c(C)nn(C)c2Cl)=O)C1)C C1(NC2(CNC(c3c(Br)cc(NC(C)=O)s3)=O)CC2)COCCC1(F)F Cc1cc(F)ccc1C(=O)N(C1CC(C#N)C1)CCNC1C2CC3C(C2=O)C13 c1(C(=O)NCC(CNC(c2cnc(C(C)C)s2)=O)C)cnc2c(c1)CCOC2 CC(Cc1ccco1)C(=O)N(C1CC1)CC1(CNC(=O)CCN2CCC2)CC1 C=CCC(C(=O)N1CCC(C(C)C(=O)NCCCOCC(C)C)C1)C(C)C C(c1ccc2c(c1)OCO2)=CC(N1CCN(C(C2CCS(=O)CC2)=O)C2CC12)=O c1(C(=O)NC)cc(C)c(C)c(F)c1.C(CC(=O)NCC1(CCOC)CC1)OCCOC N1(C(c2cnn(CC)c2C)=O)CCC2CN(C(=O)CCc3ccncc3)C2C1 N1(C(c2[nH]c(=NCC)sc2)=O)CC2CCC1CN2C(=O)C=Cc1ccc(Cl)cc1 C(CC(O)C(=O)N(C)Cc1ccc(CNC(=O)C(O)c2cnc[nH]2)cc1)SC c1(C(N2CC(CC)SCC2)=O)n[nH]c2c1CN(C(=O)Cc1c[nH]nc1C)C2 C1(NC(=O)CN2CCCCC2=O)CN(C(=O)CN2CCCCCC2=O)CC12CC2 Cc1cc(OCCCNC(C2CC(=O)N(C(C)C)C2c2cccnc2)=O)cc(C)c1 N1(C(CCC)=O)CCC2(CCN(C(=O)Cc3sc(C(C)OCC)nc3C)C2)C1 C(CC(C(=O)NCC1CCC1(F)F)NC(=O)C(CC)n1ccnc1)=CC Cc1nc(C(=O)NC2CC(C(=O)NC(C)C)C23CCC3)ccc1C#N CC1CC(c2nnnn2C2CCC2)(NCCCSC(C)C)C1 c1(C(=O)NC2C(CNC(C=CCOC)=O)CC2)coc2ccccc12 C(=O)(CCCCCCNC(C1C(C#N)C1(C)C)=O)NC(C)C(C)(C)O c1(C(N(C(C)CNC(=O)COC2(C)CCC2)C)=O)cncc(NCC#N)c1 C1(C(N)=O)CN(C(C2CCCN2C(c2ccc(C(F)F)o2)=O)=O)CCO1 CCCCC(F)C(=O)NC(c1ccnn1C)C(N1CCCC1CCCO)=O C1(CNC(C2C(C#C)C2)=O)C(C)CCCN1C(C1CCC1c1nc(S)n[nH]1)=O c1(CC(C)C)cc(C(=O)NCCCNC(C2CC(C)(C)C2)=O)no1 C1(CNC(C2CC(C)CN2C(=O)C(F)OC(F)(F)F)=O)CC(C(N)=O)=NO1 CCC(CC(=O)NCC1CC(C)N(C(c2c[nH]c(=O)cn2)=O)C1)CC(C)C C1(NC(c2[nH]cc(C#N)c2)=O)C2CCC1N(C(C1CC(=O)N(C(C)C)C1)=O)C2 CC(CN=c1ccnc(Cl)[nH]1)N(C(=O)CCN(c1ccsc1)C)C C#Cc1cncc(C(=O)N(C2CN(C(=O)CC3CN(C)C3)CCC2O)C)c1 N1(C(c2c(CC)con2)=O)C2CCC1CN(C(=O)CC(C)c1ccccc1)C2 c1(CN2CCC(NC(c3ncc(CC)nc3)=O)C2)cc(Cl)ccc1Br N1(C(CCOC(C)C)=O)CCC2OCCN(C(=O)C3=NOC(C)C3)C2C1 c1(C(=O)NC2Cc3c(C)[nH]nc3C2)cc2cccc(Br)c2[nH]1 C(c1ccccn1)=CC(=O)NCC1C=CC(NC(c2c(C(C)C)ncs2)=O)C1 C1(NC(C2(N(C)C)CCCCC2)=O)CC2CC(NC(c3ccc[nH]3)=O)C1C2 C#Cc1cc(C(=O)NC2(C)CC(C(=O)NCCC3CC4C=CC3C4)C2)ccc1C Cc1cc2c(cc1C(=O)NC1(C(=O)Nc3nccs3)CCCCC1C)OCO2 CCC(CC)C(=O)NCC(C1CCN(C(c2cc(C)n(C)n2)=O)CC1)F Cc1cnc(C(C)NC(=O)NCCc2ccc(C(F)(F)F)cc2)nc1 C1(CNC(c2nc(CCCC)sc2)=O)CC2CCC1N2C(=O)CCCSC(C)C C(C(C(=O)N1CCC(CO)C1)C(C)(C)C)NC(CCCOCCC)=O C1(CC(=O)N(CCNC(C2(SCC3CC3)CCC2)=O)CC)CCC2(CC1)COC2 Cc1csc2cc(C(=O)NCCC(C)(C)CNC(C3C(C)(C)C3(C)C)=O)[nH]c12 c1(OC)ccc(Br)c(C)c1C(=O)Nc1cnn(-c2ncccn2)c1C(=O)N(C)C C(=O)(C(CCC1CCC1)NC(=O)COC1CCOCC1)NC(C(C)C)C1CC1 CCCC(C(=O)N(C)OCC(F)(F)F)NC(C1CCOCC1(C)C)=O C12(NC(C(CSC)C)=O)CC(C)(C1)OC21CCN(C(=O)CCC[N+](=O)[O-])CC1 N1(C(C)=O)CCCC(OCC2CCCN2Cc2cccnc2C)C1 c1(C(=O)NC2C(NC(C3CN(C(C)=O)C3)=O)C2)c(C)[nH]c2ccccc12 C1(OC)CC(CNC(=O)COC2CCCOC2)N(C(=O)CCC2CCC(O)CC2)C1 N1(C(=O)C=Cc2ccc[nH]2)CCCC2(CCN(C(C3CC4C(C3)C4(F)F)=O)C2)C1 CCCC(C(=O)NC1CCCCC1CNC(C12CCC(CC1)O2)=O)OC N1(C(CCOCCOCC)=O)CCC2C(C(=O)N(C(C)CF)C)C2C1 N1(C(C=CC(C)=O)=O)CC(C2CCCN(C(c3ccc(Cl)cn3)=O)C2)C1 C(=O)(C1=NOC(C(C)(C)C)C1)NC(CNC(C(CSC)OC)=O)(C)CO c1(C(N2C3CC(CNC(CC4N(C)CCC4)=O)C2CC3)=O)ncn2ccccc12 Cc1c(-n2nnnc2C(c2cncn2C)NCC(Cl)Cl)cccc1Cl N1(C(CC2CC(OC)C2(C)C)=O)CCCC2CC1C2(C)C.c12ccsc1C(=O)N2 C1(CC(N2CC(NC(c3c(-c4cn(C)nc4)c[nH]c3)=O)C2)=O)CC2C=CC1C2 c1(C(N(CCCNC(c2c(C)coc2C)=O)CC)=O)cc2c(O)cccc2n1C c1(OC)ccc(N(C(=O)CCCCn2cc(-c3csc(C)n3)nn2)C)cc1Cl C(C(=O)NCC1CCCO1)(C1=CCSC1)N1C(CCCCC)CCC1 C1(C(=O)NCc2c(C(N(C)Cc3cc(C)on3)=O)con2)CCCSC1C Cc1nc(N2CCCC2)cc(N2CCCC(NCCC3CC=CC3)C2)n1 c1(NC(C(C)N(CC#C)C(=O)OC(C)(C)C)=O)cncc(Cl)c1 N1(C(CCCOC(C)=O)=O)CCC(C2CC(NC(=O)C(C)(C)C)C2)C1 C(=O)(C1=CC2C=CC1C2)NC(CCCOC)C(=O)NC1CC2CCCC2C1 C1(C(=O)NC(C2CCCCC2)CNC(=O)NCCC(=O)OC)(C(F)F)CCCO1 N#Cc1ccc(N2CC3C(NC(C4CCC(F)CC4)=O)C3C2)nc1 Cc1nc(O)c2c(n1)CCN(C(c1cc(Br)ccn1)C(=O)NCCCF)C2 c1(CNC(c2cc(C)n(-c3cc(C)cc(C)c3)c2C)=O)cc([N+](=O)[O-])cnc1C C1(C(=O)NC(c2ccccc2)C)COCCN(C(C2(C)CCN(C)C2)=O)C1 N1(C(C2N(C(C)C)CCC2)=O)CCC(C(=O)N(CCO)CCO)C1C(C)C C1(CCNC(c2ccc(CCC)[nH]2)=O)C(C)CCCN1C(=O)CC1CC1 C(=O)(C1CCCc2nc(C(=O)O)cn21)OCC CCC(CC(=O)NCC#CCNC(c1ccc(OC)cc1)=O)c1ccc(C)cc1 c1(C(N2CCC(CN(C(c3cc(C)ncn3)=O)C)CC2)=O)ncnc2c1CCC2 C(=O)(C1CCCc2sccc21)NC1C(NC(c2cc(COC)[nH]n2)=O)CC1 Nc1c(C(=O)NC2(CNC(c3cccc(Br)c3)=O)CC2)cc(F)cc1F c1(C(=O)NCC)nc(CO)oc1C.c1(C(N(CCOC)C(C)C)=O)cc(C2CC2)[nH]n1 C1(NC(Cn2c(C)ncc2)=O)CN(C(C2CCCC3(CC3)C2)=O)CC2(CC2)C1 c1(CCN(CC(C)O)C(=O)NCCC2(C)CC2(F)F)ccccn1 CC1(C)CCC(C(=O)NC2CC3CC2N(C(=O)C2=CCCC2)C3)OC1 CC1CCOCC1C(=O)NCc1ccc(C(=O)NC2CCN(C(C)(C)C)C2)cn1 N1(C(c2c(C)nc[nH]2)=O)CCSCC1CCNC(c1cc(C#N)no1)=O c1(C(=O)NCCN(C(C2C(C)(C)C2(F)F)=O)CC2CC2)cncc2c[nH]nc12 c1(C(N2CC(CC)N(C(C3CC(O)CN3C)=O)CC2)=O)ccc(F)c2ccoc12 C1(NC(CC(C)O)=O)CN(C(=O)CCc2cccnc2F)CCC1CO C(c1cccc(F)c1)=CC(=O)NCCC(C)CCNC(=O)COC(F)(F)F c1(NC(C)CCc2cnccn2)cc(NCCCS(C)=O)ncn1 CCC(C#N)(CC)C(=O)N1CCC(O)(CNC(=O)CC2CCCC(C)(C)C2)CC1 C1(NC(C(C)CC2CCC2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1n1cccn1 C1(C(=O)O)CCC(C(F)(F)F)CN1C(=O)Cn1nc(C(F)(F)F)oc1=O C#Cc1ccccc1CC(=O)NC1(C2CCCN2C(=O)C(C)SC)CC1 C(=O)(C1CCSc2ccccc21)N1C(CNC(c2c(F)ccc(C)c2)=O)CC1 c1(CNC(=NCCOC)NC2C(F)(F)C23CC3)c[nH]c2cc(Cl)ccc12 N1(C(CN2CCN(C(CC(CC(=O)OC)C)=O)CC2)=O)CCC(C2CCOC2)C1 C(=O)(CCCN(C)C(C1CCC1(F)F)=O)N1CC(COC)C1 C(=O)(C(F)(CNC(C1CC(C)(C)C1)=O)C(C)C)NC(C(CC)C)C C1(CC(N2CCC(C(C)NC(c3cn(C4CC4)nn3)=O)C2)=O)CCCC(C)(C)C1 c1(C(=O)NC2CCCC(NC(c3c(C)n(C)cn3)=O)C2)ccc(C(C)C)c(F)c1 N1(C(C2C(C)C2)=O)CC2CC(C1)CN(C(c1cccc(C3CC3)n1)=O)C2 C(=O)(C(F)(F)C(O)C(C)C)N1C2CN(C(c3cc(CC(C)C)on3)=O)C(CC2)C1 c1(C(=O)NC2CCN(C(C(CC)Oc3ccccc3F)=O)C2)cc(Cl)cnc1O c1(CNC(c2nc(C(=O)OC)oc2)=O)nn(C)cc1CO.C12(CCC1)C(=O)C=CC2 c1(C(=O)OC)ccc(S(=O)(=O)N2CCC3(CN(Cc4cnn(C)c4)C3)C2)n1C C(=O)(CCCCC(N)=O)NC(C(=O)NCC1CC(C(C)(C)C)C1)CO N1(C(C(C)OCC)=O)CCCC(C(=O)N(CC(C)C#N)CC2CC2)CC1 CC1(C)CCC(CC(N2CCCC(CC(=O)NC3CC4CCC3O4)C2)=O)O1 C1(C(=O)OCC)C(O)C(O)CN1C(c1ccn(-c2ccc(Cl)c(Cl)c2)n1)=O C1(C(=O)NC2CCC(NC(c3cc[nH]c3C3CCC3)=O)C2)(COC)CCOC1 C1(C(=O)OCC)CCC(C(=O)N(C)CCOCC)C1.c1(C(=O)N)cnn(CC(C)C)n1 Cc1cc2[nH]c(C(=O)NC(CNC(c3ccc(S(C)=O)cc3)=O)C3CC3)cc2s1 C#Cc1cn(C)nc1C(=O)NC(CC(F)F)C(=O)NC1CCCCC1OC C1(CC(=O)N(CCC(=O)OC(C)(C)C)CCSC)C2CCC(C2)C1N.CC(C)(C)O Cc1csc2cc(C(N3CCN(C(C4(C)COCCO4)=O)CCC3C)=O)[nH]c12 c1(C(=O)NC(CCNC(CC(CCC)C)=O)C)cc2cnn(C(C)C)c2nc1C c1(C(=O)OC)ccc(Cn2cc(-c3nccc(C)n3)nn2)cc1CC1CCC1 Cc1c(C(N2CCN(C(C3CCCS3)=O)CC3(CC3)C2)=O)sc2ncnc(N)c12 CCC(CC(=O)NC1CCC(NC(=O)C(C)(C)N2CCOCC2)C1)C(C)(C)C C(=O)(C(C)(C)C(C)(F)F)NC(C(=O)NC(C)Cc1nn[nH]n1)Cn1ccnn1 N1(C(C2CC3(CC(NC(c4c(C)n(C)cn4)=O)C3)C2)=O)C(C)CCC1(C)C N1(C(C2(CC(C)C)CCCC2)=O)CCC(NC(c2cc(CO)ccn2)=O)C(O)C1 c1(SCC(=O)NCC2CC(NC(COCC=C)=O)C2)cc(C)ccc1C N1(C(=O)C(c2cccc([N+](=O)[O-])c2)O)CC2(C1)CN(C(C1(CF)CC1)=O)CCO2 N1(C(CCOC)=O)CC(c2ccccc2)(CNC(=O)CCCSC)C1 C1(C(N(C)CC2CCN(C(=O)CCC3CCCC3)C2)=O)CC12CC(F)(F)C2 c1(CNC(C2C(C)OCCO2)=O)ccc2c(c1)CN(C(=O)CCCC#N)C2 c1(C(N(CC(C)NC(C(CCC)C#N)=O)C)=O)cc2sc(C)cc2[nH]1 c1(CC(N2CC(C)C(C)C2)=O)ncn2c1COCC2 C1(C(=O)OCC)C2CC(C2)N1C(c1cn(CCN(CCO)CCO)cn1)=O c1(C(=O)NCCCC2OCCN(C(C3(C)CC3)=O)C2)n[nH]c2c1CCCC2 C12(NC(N3CCN(C(C(C)(C)C(F)F)=O)CC3)=O)CCC(CC1)C2(C)C O=S(=O)(c1ccc(NCC2C=CCCC2)nc1)NCC(O)COCC(F)(F)F C#CCC(C)(C)C(=O)NCC1CC1NC(=O)Cc1cc(Cl)n(C)n1 C1(C(=O)NCC(CNC(c2cc(C)c(=O)n(C)c2)=O)C)CCc2n[nH]cc2C1C C1(CNC(C(C)OCC#C)=O)CN(C(c2ccn(C)c2CC)=O)CCO1 C(=O)(C1=CC2C=CC(C1)C2)N1CCOCC(C(=O)NC(C)CO)C1 C=C(Br)CN=c1nc(N2CCc3nn(C)c(=O)cc3C2)c2c([nH]1)CCC2 C(N=c1[nH]c2c(c(=NCC3C4CCCC34)[nH]1)COCC2)c1c(C(F)(F)F)ocn1 C1(NC(c2ccc(C(F)F)o2)=O)CCN(C(=O)C=Cc2ccoc2)CC1F N1(C(C(CCCC)(C)F)=O)CC(CNC(c2cnc(S)n2C)=O)OC2(CCC2)C1 N1(C(C2CN(CC)C(=O)C2)=O)CCCC(C)(NC(=O)C(=Cc2ccco2)C)C1 N1(C(Cc2c(C)cco2)=O)CC(C)CCC1C(=O)NC(c1ccc(Cl)cc1)C CC(C)(O)C#CC(=O)N1CCC(N2CCN(C(C3OCCOC3(C)C)=O)CC2)C1 C(c1ccc(C)cc1)=CC(=O)NCCC1CCN(C(C2(OCC)CCC2)=O)C1 C(=O)(CCCCC(C)(C)C)N1CCC(NC(CS(N2CCC(C)CC2)(=O)=O)=O)C1 CC(C)CC(C(=O)N(CC(C)NC(C12CCC(C(F)F)(CC1)C2)=O)C)C(N)=O Cc1[nH]c(C(C)(C)C)cc1C(=O)NCCC1CCN(C(=O)C(C)C2CC2)C1 N1(C(c2cccc(CCC)c2)=O)CC2CC1CN2C(c1cn(C)ccc1=O)=O C123CCC(N=CNC(CO)=Nc4cccnc41)(CCC2CC)CO3 C1(C(C(N2C(C(=O)NCC=CCCC)CSC2)=O)C)CN(C(C)=O)CCO1 c1(OC)cc(OC)c(C(=O)NCC(F)CNC(c2nccc(C)n2)=O)c(N)c1 C(=O)(CC(=O)c1ccccc1)N(C(Cc1cccnc1)C(=O)O)CC(C)C c1(CCC)nc(C)c(C(N2CCOC(CNC(=O)CCn3cncn3)C2)=O)s1 N1(C(c2ccc3c(c2)COC3)C(=O)NCC)C2CCC1CC(CO)C2 CCCCCC(=O)NCc1ccc(CNC(C2CCCN2C=O)=O)o1 c1(C(=O)NC2CC(F)(CNC(C(C)SCC)=O)C2)c(F)cc(COC)cc1F N1(C(C(C(C)C)n2cccc2)=O)CCC2(CCN(C(=O)C(F)(F)C(F)F)CC2)C1 N1(C(c2cc(CNC(C(C)NC(CC)=O)=O)no2)=O)CC2CC=CC1C2 C1(CC(=O)NCC(N2CCN(C(C3(C)CC(C)C3)=O)CC2)C)CCCC(C)(C)C1 CC1CCn2cc(CNC(=O)NCC34CCC(C(=O)O)(C3)OC4)nc2C1 c1(OC(=O)Cn2nc(C(COC)=O)c3c2CCC3)cccc2c1CNC2=O N1(C(c2cccc(NC(N)=O)c2)=O)CCCC(C2CC2NC(C2(O)CCC2)=O)C1 c1(C(c2nnnn2NCC#N)SC)ccc(Nc2cccc(OC3CC3)c2)nc1 c1(NC(c2n(CC(=C)C)nnn2)C2(CC)CCCC2)ccc(C2(C)CC2)cc1 C(CC(=O)NOCc1cc(-c2ccccc2)ncn1)S(CC)(=O)=O c1(C(=O)NC2(C(NOCCCC=C)=O)CSC2)c(C)nsc1N c1(C(N2CC3(C(NC(C4CC45CC5)=O)CCC3)C2)=O)ccc2nc(S)oc2c1 C1(C)(NC(C2CCN(C(CC)=O)C2)=O)CCN(C(c2cc(OC)cs2)=O)C1 C(CCNC(=O)CC1CN(C(=O)OC(C)(C)C)CCO1)(C(C)C)OC C1(CNC(CC(CNC(=O)CCc2nc(=N)[nH][nH]2)OC)=O)CCCC(C)(C)C1 CC(C)(O)C#CC(=O)NC1CC1CNC(C1CCCC(C2CC2)O1)=O N1(C(C2(COC)CC2)=O)CCC(n2cc(C3(C(=O)OC)CCCC3)nn2)CC1 C1(C(F)(F)F)(C(=O)NCC(C)(C)NC(C2C(CCC)CCC2)=O)CC(F)(F)C1 N#Cc1cccc(C(N2CCC(CC(=O)NCC3CCCO3)C2)=O)c1 C1(C(=O)NCCN(CCC)C(C2CCCC(=O)O2)=O)CN(CP(C)(C)=O)C1 C(=O)(C(CC(C)C)OC)N1CC(C(=O)NC(C#C)C(C)(C)C)OCC1 C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCC(NC(C(CCC)CC)=O)CC1 C(CCCCC(=O)NC1CC(CCO)C1)c1cn(CC(CSC)(C)C)nn1 C1(C(=O)NCCOC(C)C)CC2CC2N1Cc1ccc(Br)s1 c1(C(CC)C)ccc(C(=O)N(CCCNC(C23CCC(C2)OC3)=O)C)cc1 N1(C(c2c(F)c(F)c(NC(C3C(C)C3)=O)c(F)c2F)=O)CCc2cccc(Br)c2C1 CC(C)C(CCC(=O)NCC(CC1CC1)CO)NC(=O)CCC1(C)N=N1 CC1(C)CN(C(c2cc(N(C)C)ccc2N)=O)CCC1NC(c1cnsc1)=O C1(NC(CC=CC)=O)CCC(C)N(C(c2cccc(N(C)C)n2)=O)C1 N1(C(=O)CCC2=CCSC2)CC(CC(N2CCC2C2CCCCC2)=O)C(CO)C1 CCC(C)C(O)C(C)C(=O)NCC1CC(NC(=O)C(C)(F)C(=O)OC(C)(C)C)C1 N1(CC2(OCC)CNC2)CCC(N(C)C)CC1.OC C=CC1(CC(=O)NC2CCCCC2NC(C2CCOC2C2CC2)=O)CCOCC1 C1(N(C(COCC(=C)C)=O)C)CCCN(C(=O)CCc2scnc2C)C1 c1(NC(C2(F)CCN(C(Cc3cc(C)on3)=O)CC2)=O)ccc(F)c(Cl)c1 N1(C(C(C)c2cccs2)=O)CC2N(C(C3C=CCC3)=O)CCC2(C)C1 c1(SCC23CCCC(C)(C2)CO3)ccc2[nH]cc(C(=O)CC3CCCC3)c2c1 c1(C(=O)NC2C(NC(c3cc(C)c(C)nc3)=O)C2)ccnc2ccc(F)cc12 O=C(C1NCCn2nccc21)NC1CC(N2CCCC2)C1 Cc1cc(NCC2CCN(C(c3cc(C4CC4)on3)=O)C2)c(C#N)cc1[N+](=O)[O-] C1(OC)CN(C(c2ncc[nH]c2=O)=O)CC1NC(c1c(Cl)nsc1Cl)=O CCS(=O)(=O)CC(=O)N(CCC(=O)NCC(C)(C)C(C)O)C C(C(=O)N=c1ccn(C(C)(C)C)[nH]1)(c1cccnc1)NC(C(CCCC#C)C)=O C1(NC(CNC(CCC)=O)=O)CC2CC(C1)N(C(c1nnn(C)n1)=O)C2 CC(C)CC(Cc1ccccc1)C(=O)N1CCN(C(c2ccc(CO)s2)=O)CC1 Cc1nc(C(N2CCC(C)(O)C2)C(=O)NC2COC2)c(C)n1C Cc1cnc(C(=O)NC2C3CN(C(C45CCC(CC4)O5)=O)CC23)cc1Br C1(NC(C2(C)CCOCC2)=O)CCN(C(c2cc(C3CCCC3)no2)=O)CC1F N1(C(CCN(C2CC2)CC)=O)CCCN(C(=O)C=CCCCCC)CC1C c1(CNC(C2(C(F)(F)F)CCC(NC(=O)OC(C)(C)C)C2)=O)cc(Cl)cnc1C C(=O)(CCN(OC)C(=O)Cc1cc(O)ncn1)NCC1CN(C(C)=O)C1 N1(C(C(C)SCCCC)=O)CCC2(CCCC2CNC(C2(N(C)C)CC2)=O)CC1 N1(C(C(CC)COC)=O)C2CCC1C(NC(=O)Cc1cc(F)ccc1Cl)C2 c1(C(=O)NC(CNC(C(CC)(C)COC)=O)(C)C(C)C)cc2ccncc2[nH]1 C1(NC(c2c(C)nns2)=O)COCCC1NC(c1ccc(C(C)(C)C)[nH]1)=O Cc1cc(F)c(C(N2CCN(CC(C)C)CC2)=O)cc1-c1cccnc1C N1(C(C(COC)OC)=O)CCCC(CCOC)(NC(C2(CCO)CC2)=O)C1 c1(CC)ccc(C(=O)NC2CC(C)(NC(c3nc(CC)ncc3Cl)=O)C2)cc1N C1(CC)CN(C(c2ccc(COC(F)F)cc2)=O)CC(CC(=O)O)O1 Cc1cc(CNC(C2COCC2C(N)=O)=O)nnc1C.C12CCCCC1C(=O)NC2 Cc1cc(=O)c(C(=O)NCC(C)CNC(=O)CC2CCC23CCC3)cn1C CC(C)C(C#N)C(=O)NCC1CN(C(=O)C(C)(C)c2ccn(C)n2)C1 CCCCCC(F)C(=O)NC(C)CCC(=O)NCC(O)C(F)(F)F n1(CC)nc(C)c(C(=O)NC2CC(O)(CNC(=O)C(=O)NC(C)C)C2)c1Cl c1(CC(C)NC(=O)Nc2ccoc2SCC2CC2)cn(C)c2ccccc12 CCCCC(C(=O)NCC1CCOC(C)C1)NC(=O)CNC(=O)CN(C)C c1(CC(=O)NC(CCCC)CNC(=O)CC(C)CF)ccc(S(N)(=O)=O)s1 N1(C(C2(F)CN(CCCCC3C(C)C3)C2)=O)C(C)CCC1C n1(CC(N2CCC(CNC(c3c(C)oc(C#N)c3)=O)C2)=O)nc2c(n1)CCCC2 Cc1cc(C(=O)NC2CCC2NC(C2(c3ccccc3)CCOC2)=O)nn1C C=CCC(CC=C)C(=O)NC1(C2CN(C(c3ccc(F)cc3N)=O)C2)CC1 c1(C(=O)NCC(CC)N(C)C(c2cn(C)cn2)=O)cccc2cnn(C)c12 C(CN=c1cc(C(F)F)nc[nH]1)C1N(C(C(CC)n2ccnc2)=O)CCC1 c1(C(N2CCC(CN(C(=O)CCC(F)(F)F)C)C2)=O)ccc(F)c(F)c1F N1(C(c2ccc(C)cc2)=O)CCN(C(=O)CC2CC(C3CC3)=NO2)C(CCO)C1 C1(CNC(C(C)CN(C)C)=O)CN(C(=O)Cc2nncn2C)C2COCC2O1 c1(CCNC(C2CCN(CC(C(C)(C)C)O)CC2)=O)cccc(F)c1F c1(C(=O)N(C(c2ccccc2)C(=O)NCC(F)(F)F)CCO)ccnn1CC(F)F CC(CN=c1nc2c(cnn2C)c(NC2CCCC3(CC2)CC3)[nH]1)c1nccs1 n1(CCC(=O)NC(CC(C)NC(C=CSC)=O)C)c(S)nc2ccccc2c1=O c1(OC)cc(C(N2CCC(CNC(=O)CCCCC#N)C2)=O)ccc1Cl c1(C(=O)NC2CCCC(NC(C3CCOC3C(F)(F)F)=O)C2)csc2nnsc12 Cc1ccc(F)cc1C(N1C(CNC(=O)Cc2ccccc2F)CC2CC12)=O c1(CC(=O)N(C)CCN(C)C(C2CCCOC2)=O)ccc2c(c1)COCC2 c1(CN(C(=O)NCC(C(C)OC)(C)C)C2CC2)cccc(C#N)c1 C(=O)(CC(C)(C)CC(C)=O)N1C(CCNC(C=C(C)C2CC2)=O)CSCC1 c1(C(=O)NCC(C)CN(C(=O)Cc2cnnn2C)C)cccc(C#CCO)c1 N1(C(CC2(COC)CC2)=O)CCCCCCC1C(=O)NC1CC(O)C(O)C1 C1(C(=O)NC2(CCCC)CC2)CC2CCN(C(C3CCC=CO3)=O)CC12 N#Cc1c[nH]c(C(N2CCC2CN=[N+]=[N-])=O)c1.N12CC(C1)CC2=O N1(C(Cc2c(C)scc2)=O)CCC(C)C(NC(c2c[nH]nc2C2CCCO2)=O)C1 C1(NC(C2(C#C)CC2)=O)CCC(C)N(C(c2scnc2CC)=O)C1 N1(C(=O)OCC)CSCC1C(=O)NC(C)(C)CN(C)C(c1sccc1Cl)=O c1(C(=O)OC)cnc(Cl)cc1NC(C1(C)CCN1c1cc(OC)ncn1)=O CC1CCN(C(=O)CSc2ccc(F)c(F)c2)CCC1(F)F C(C(C(=O)NCC1COCCN1C(=O)Cn1cccnc1=O)C(C)(C)C)N(C)C C1(C(=O)NC(CC)CCOC)(CC)CCN(C(=O)Cc2cc(C)on2)C1 C1(NC(CCCNC(C)=O)=O)CCN(C(C2CN(C(N)=O)C2)=O)C(C)C1 c1(OC)ccc2c(c1)C(Nc1ccc(Cl)c(C(F)F)c1)CC2 C1(NC(c2c(CCC)cccc2)=O)CCN(C(=O)C(C)(C)CCOC)CC1CC C1(C(=O)NC2CCCCCC2NC(c2n(C)nc(CO)c2)=O)CC2(CCOC2)C1 Cc1cscc1C(N1CCCC1CC(=O)N1CCC1C(N)=O)=O C12CN(CCO1)C(=O)C(C)(CC)O2.n1(CC=C)cc(C2(C)CNC2)nn1 c1(OC)ccnc(C(=O)NCC2(NC(c3ncoc3Br)=O)CCC2)c1 O=C(C1=COCCO1)NCC1COCC1NC(C1CCCC12CCC2)=O N1(C(C2CCN(C)CC2)=O)CCC2CN(CC3CCC3)CC2CC1 C1(CC(=O)NC(C)COCC(F)(F)F)COCCN1C(=O)C(C)C(F)F c1(C(N2CC(NC(c3cnn(C)c3Br)=O)C3(C2)CC3)=O)cc(N)c(Cl)c(O)c1 N1(C(c2ccc(OC)c(F)c2)=O)C2CCC1CN(C(C1CCOC1C)=O)C2 N1(C(C2(CCNC(C(CC)SC)=O)CCC2)=O)CCC12CCCC2 c1(SCC(N2CC(OC)C(NC(c3coc(Cl)n3)=O)C2)=O)ccc(C#N)cc1 c1(C(=O)NC)ccc(CSc2ccc(F)cc2)cc1.C12CC(C1)NC(=O)N(C)C2 N1(C(CC(C=C)(C)C)=O)CCC2CN(C(=O)C(C(C)C)NC(=O)OC)C2C1 Cc1nc(N2CC(NC(=O)CC(C)C3CCCO3)CC3(CC3)C2)cc(C#N)n1 C1(C(N(C(C)COC)CC=C)=O)CCN(C(=O)c2cccn2C)O1 c1(OCC)oc(C)nc1C(=O)N(CC(C)NC(=O)C(C)Cc1c(C)noc1C)C C1(NC(=O)Cn2cc(C(N3CCCC3)(C)C)nn2)CCC(c2ncc[nH]2)CC1 C1(CC(C)C)(C(=O)Nc2ncc(-c3ccccn3)s2)CCNC1 N(C1CN(C(C2(CF)CC2)=O)Cc2ccccc21)C(CC=CCC)=O C(=O)(C(C)(C)CC(C)C)NCC(CC)NC(=O)C(N1CCCC1)C1CC1 C1(NC(c2cnco2)=O)CCCC12CN(C(c1cccnc1-n1ccnc1)=O)C2 c1(-n2cc(CCNC(C3C(C(C)C)CCC3)=O)nn2)ccc2c(c1)oc(=O)n2C C1(CNC(C(=O)N(CC(c2ccccc2)CC)CC)=O)CCC(=O)N1C N1(C(C(C=C)c2ccccc2)=O)CC2C(C(=O)N(CC(C)(C)O)CC(C)C)C2C1 c1(CCC(=O)N(CC(C)N(C)C(C2C3COCC23)=O)C)nc(C2CCCC2)no1 c1(S)cc([N+](=O)[O-])ccc1N.C#CCCCN(C(=O)Cn1ccnc1)C Cc1c(C(N2CCC(CNC(=O)C3=NOC(C)(C)C3)C(C)C2)=O)cc(N)cc1O C(CCC(F)(F)F)(C(=O)NCC1CCC(F)(F)CC1F)NC(C)=O CCC(C)C(O)C(=O)NCc1cccc(CN(C)C(c2cnc(CC)nc2)=O)c1 Cc1cc(F)c(NC(=O)CC(C(C)C)NC(=O)Cc2ccoc2)cc1F Cc1c(NC(=O)C(N2CCCC2C(=O)Nc2ccnc(F)c2)=O)cccc1F C1(NC(C(C)OCC)=O)CCCCCC1C(=O)NCC(C)(C)N1CCCC1 C1(C)(C(=O)NC2C(CNC(C(C)=CC3CC3)=O)CCCC2)CCC(F)(F)C1 Cc1nc(C)c(C(C)NC(=O)CCN(C(c2ncccc2C)=O)CC2CC2)[nH]1 C(=O)(C1CCCc2nn[nH]c21)NCCC(CNC(C(C)SC)=O)(C)C N1(C(=O)COCCN(C)C)CC2(CCCN(C(c3cnc(C4CC4)o3)=O)C2)C1 c1(-n2cc(SC(C)C(C(=O)O)OCc3ccccc3)nn2)ccc(F)c2occc12 C1(NC(c2cc(C)n(C)c2)=O)CCN(C(C2CCOC2)C)C(C)C1 N1(C(C(C)C#N)=O)CCC(C)(C)C(NC(c2cccc(Br)c2F)=O)C1 C(=O)(C1CCCc2nn[nH]c21)N1C(CCNC(C=CC=CCC)=O)CSCC1 CC1CN(C(C2CCCN2C(c2cccc(C#N)c2)=O)=O)c2ccc(F)cc2O1 c1(OC)c(C(N2CCN(C(C3CC4C=CC3C4)=O)C(C)C2)=O)cccc1Br c1(CNc2ccc(NC3CCCN(C)C3c3cccs3)cc2)noc2c1CCCC2 c1(C(N2CC(C(C)(C)O)(C(=O)NCc3ccc(CC)o3)C2)=O)cc(O)ncn1.C=CC C1(NC(CC(c2ccc(F)cc2)C)=O)CCC(Nc2cc(F)ncn2)CC1 n1(C(C)C)nnc2c1CCN(C(C1CC(C3CCNCC3)C1)=O)C2 c1(NC(C2(F)CCN(Cc3nccc(OC)c3)CC2)=O)cccc2c(C)[nH]nc12 C(=O)(CCCS(C)(=O)=O)NCC1CCN(c2ccc(C(C)=O)cc2)CC1 N1(C(c2ccc(OCCCC)cc2)=O)CCC(CCNC(C)=O)C(Br)C1 CC1CCN(C(=O)Cc2ccc3c(c2)CC3)CCS1 C1(C)(C(=O)NC2C(OC)CN(C(C(CC)NC(N)=O)=O)C2)CC2CCC1O2 N1(C(=O)Cc2ccon2)CC2(C(N3CC4C=CC4C3)=O)CC1CCO2 c1(C(N2C(CNC(=O)CC34CCC(CC3)C4)CCCC2)=O)cccc2c1OCC2 CC1(CNC(=O)C=Cc2ccccn2)COCCN(C(c2ccsc2Cl)=O)C1 C1(CC(=O)NCCCNC(=O)C=Cc2cc[nH]n2)CC(O)C12CCC2 C1(CCC(=O)NCCNC(C2(CCCC)CCCC2)=O)CCc2cnn(C)c2C1 CC1CCCCC1(CNC(c1cc(F)cnc1O)=O)NC(=O)C=Cc1cocn1 N1(C(CC2(NC(C)=O)CC2)=O)CCCC12CCN(C(c1snnc1C)=O)CC2 C1(NC(C(n2ncc(C)c2)C)=O)CC2(C1)CC(NC(C1CCC(F)C1)=O)C2 CC1OC(C)C(C(N2CCN(C(=O)CCCCF)CC2CCO)=O)C1C CC(C)C(C(=O)NC(C)CCNC(=O)C=Cc1cocn1)n1cnnc1 c1(CNC(C=C(COC)C)=O)ccc(CNC(c2cn(C)nc2OC)=O)c(F)c1 Cc1cc(S(N)(=O)=O)oc1C(=O)NC1CC2CCC(C1)N2C(=O)CCC1CCC1 C1(CC#C)(C(=O)NCCn2ncccc2=O)CCN(C(=O)COCCF)C1 c1(C(=O)NCC2(CC)CN(C(c3cccc(=O)n3C)=O)C2)cn2ccccc2n1 C(=O)(C(C(=O)NCC#CCNC(=O)CC(c1ccc(F)cc1)C)OC)OCC C1(CC(=O)NC(C(C)F)C)COCCN1C(=O)CCc1ccn(C)c1 c1(C(N(C2CC(NC(c3ccc(NC(C)=O)s3)=O)C2)C)=O)cnc2ccnn2c1 c1(C(N2CC(C#N)C(NC(c3ccc(Br)c(Br)c3)=O)C2)=O)cccc2c1CCC2 Cc1cc(O)ccc1C(N1CCC1C(=O)Nc1c(Cl)cccc1Br)=O c1(NC(CCC2CC(NC(=O)CC3CSC3)C2)=O)ccc2c(c1)OCC2 N1(C(C(CC)C)=O)CCCC(CCNC(=O)COc2nn(C)cc2Br)CC1 CC(CCC(C)(C)C)C(=O)NCC1CN(c2nnco2)CCC1(C)C C(CCCC(=O)NC1C=CC(C(=O)NC2CC2(C)C(=O)OCC)C1)SCC=C N1(C(c2sc(Br)nc2C)C(=O)NCCOCC)CCN(C)CC12CCCCC2 N1(C(C(C)=C2CCC2)=O)CC(C)C(NC(c2ccc(C)c(C)n2)=O)C(C)C1 C1(C(=O)NC(CCC)C2CCC2)C(CC)CCN1C(=O)CC1CSCCO1 CCC(C)C(=O)N(C(C)(C(=O)NCCC(C)CO)C1CC1)C CC1OC2(C)CC1(C(=O)NCC1(C(N)=O)CN(C(c3cc(C(N)=O)cs3)=O)C1)C2 C1(C2CC2)(CNCC(=O)Nc2cc(F)cc(F)c2)CC=CC1 CC1CC(F)(F)CCN1C(=O)C(CNC(c1ccc(N)cn1)=O)C(C)(C)C N1(C(c2c(C)con2)=O)CCC(SCC(=O)N(c2cccc(O)c2)C)CC1 C(=O)(C(O)CC(C)(C)C)N(CCN(C(=O)CCc1ccc(F)cc1)C(C)C)C c1(C(=O)NCC(N(C(Cn2c(C)nnn2)=O)C)C2CC2)c(N)ccc(F)c1F C(CCC(=O)NOOCOC)(C(C)C)N(C(C1CCCN(CC)C1)=O)CC C1(CNC(C(c2scc(C)n2)C)=O)(NC(=O)CC2OCCC2C)CCCCC1 C1(SCC)CCN(C(=NCC(C)C)NCC(C(C)C)OC)C1 Cc1cc(=N)[nH]cc1C(N1CCC(O)(C(C)CNC(c2cnn(C)c2Cl)=O)C1)=O Cc1ccc2c(C(=O)NC3CN(C(=O)CCc4ccn(C)n4)CC3F)n[nH]c2c1 c1(NC(C2(CNC(=O)NCC3(C4CCCO4)CCCC3)CC2)=O)cccc(Cl)c1 C12CCCC1NC2=O.C(C(C)C(F)F)NC(COCCCC)=O CC(O)CC(C)CN=c1[nH]c(=NCc2ccc(OC(C)C)c(Br)c2)[nH]c2cc[nH]c12 C1(O)(CNC(C2CCCN(C3C(=O)NCCC3)C2)=O)C2C3CC4C5C3CC2C5C14 N1(C(CC(=O)NC)=O)CCN(C(C2(COC)CCCCC2)=O)CC1CC(F)F N1(C(=O)NC(c2cn(-c3ccccc3Cl)nn2)CC)CCN(C)CC1C(C)C C1(C(=O)NCC(CCC)(C)O)CN(C(=O)C(OC)OC)CC(C)(C)C1 C=CC1OCCC1C(=O)NCC(c1cccc(C)c1)NC(=O)CNC=O N1(C(CC(C)OC)=O)CCCC(NC(=O)Cn2ncc(Br)n2)C1 C(=O)(C1=CC2(CCOC2)C1)NC(C1CN(C(=O)CC2(O)CCCCC2)C1)C C(c1ccccc1Cl)=CC(=O)NC(C)CCCCNC(C1CCCN1C=O)=O C(=O)(CCCCCCN=[N+]=[N-])N1CCC(CNC(CC(CCC)O)=O)CC1 c1(C(N(C2CCC(NC(CN(C)C(N)=O)=O)C2)C)=O)cccc(-n2ccnn2)c1 c1(C(=O)NCC2OCCN(C(CCC)=O)C2)nn(C)c(C(F)(F)F)c1Cl C1(CNC(c2c(CC)c[nH]c2)=O)CC(C)CN(C(C2CCC(C(C)C)CC2)=O)C1 C1(NC(CCCOC)=O)C(C)(C)CN(C(c2nc(OC)c(C)s2)=O)CC1(C)C c1(C(N(CCC)CCNC(c2ncc(F)cc2C)=O)=O)cc(S(C)(=O)=O)co1 c1(C(=O)NCC2CC2NC(C2CC2(Cl)Cl)=O)cc(Cl)ccn1 c1(C(=O)NC2C(NC(C3N(C)C(=O)CC3)=O)CC2)ccc2nnn(O)c2c1 CCC(C(=O)NCC1(C(=O)NC(C(F)(F)F)C2CC2)CC1)n1cncn1 c1(C(=O)NCCCOCCNC(CCC(C)OC)=O)ccc2c(c1)CCCC2=O C(=O)(CCC(CF)CF)N1C(CC)C(CNC(C2NCC2)=O)CC1.C(=O)OC c1(OCc2ccccc2)cc(NC2CC(NC3CCC3)C2)ncn1 CCCCC(C(=O)NCCCCC1CC1)NC(c1cnc(C2CC2)o1)=O c1(C(N(CCCCNC(C(CC)(C)F)=O)C)=O)cnn2c1NCCC2C(F)(F)F c1(C2(C(N3CC(NC(COCC(=O)OC)=O)C(C)C3)=O)CC2)ccc(C)c(C)c1 Cc1cc(C=CC(=O)NCC(O)CNC(C2CC2C(F)F)=O)ccc1OC(C)C C12(C)CCC(CC1)NC(=O)N2Cc1ccccc1Cl.Cn1nnnc1SC1COC1 c1(C(=O)NCC2N(C(C(CC)SC)=O)CC3(CC3)C2)cn(C)c(=O)n(C)c1=O C1(CNC(C2CCCC2)C)CN(C(=O)OC(C)(C)C)CCO1 c1(C(=O)NC(CNC(C2(CC#C)CCCOC2)=O)C)ccc(C(C)(F)F)nc1C C1(NC(C2(CC)CCC2)=O)CC2CCC1N(C(c1c(C)cc(C)nc1O)=O)C2 N1(C(C(C)NS(C)(=O)=O)=O)CCc2cc(CNC(C3CC3C(F)F)=O)ccc2C1 Nc1c(C(=O)NCC(CO)NC(=O)C=Cc2ccoc2)ncc2ccccc12 N1(c2cc(C)nc(CO)n2)CCC2CC(NC(c3cc(O)nn3C)=O)CCC2C1 n1(CN(CC(C)(C)CNC(=O)OC(C)(C)C)C)cc(CO)cc(C(=O)O)c1=O C1(N(C(=O)CC23CC(C2)C3)C)CCN(C(C2(C(F)(F)F)CCC2)=O)CC1 C(=O)(C(CC)CCCC)NCC(N1CCN(C(C(CCCC)O)=O)CC1)C c1(C(=O)NC(CN(C(c2ccc(OCC)cc2)=O)C)C)cncc(C)c1Cl N1(C(c2nc(C)nc(=N)[nH]2)=O)CC2CN(C(=O)OCC(C)(C)C)CC2(C)C1 c1(OC)ccc2cncc(C(=O)NCCCOCCNC(C3(F)CCC3)=O)c2c1 CCCS(=O)(=O)C(C)C(=O)NC(C1CCCN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1)C N1(C(=O)Cc2cncnc2O)CC2CCC(C1)N2C(C1CCSC1)=O C(=O)(CC(C)(C)C#N)NCC(CN(C(=O)C(F)C1CCOC1)C)(C)C C(=O)(C(CC(=C)C)OC)NC(CC#C)C(=O)N(C(C)CC(N)=O)C N1(C(C(CC)SC)=O)CCC(O)C1C(=O)NC(c1ccns1)C C1(CNC(=O)C2=CCC2)CCC2(CN(C(c3cc4ncccn4n3)=O)C2)O1 c1(CC(C)C(=O)NCCOCCNC(C2(CO)CCC2)=O)ccc([N+](=O)[O-])cc1 CC1CCCC1N=c1nc(N2CCC3(CC2)C(F)(F)C3(F)F)c2cccc(F)c2[nH]1 CC1CCCCN1CC(=O)NC1CC(C)(NC(C2CC2C(F)F)=O)C1 c1(OC)ccc(C(=O)NCC2CC(O)(CNC(=O)C(C)(C(C)C)OC)C2)c(O)c1 S(=O)(=O)(c1ccc(N2CCn3c(C)cnc3C2)c(F)c1)NC1(CCOC)CC1 N#Cc1cncc(CN2CC(NC(c3ccccc3)=O)C2)c1 CCC(C)C(O)C(=O)N1CCC(C)(NC(C2CCN(C)CC2)=O)CC1 c1(C(C)C)cc(C(=O)NCC2(NC(=O)C(C)(O)C3CCC3)CCC2)ccc1N CC1CN(C(C2(C3CC3)CN(C(=O)C=Cc3cscn3)C2)=O)CCC1CO c1(CNC(COC2CC(NC(C(COC)C)=O)C2)=O)ccc(Cl)c(C)c1 CC1C(=O)CC1C(=O)N(CCCN(C)C)CCNC(=O)CC1(C(F)(F)F)CC1 c1(CC(=O)NC(CC)CN(C)C(c2ccon2)=O)ccc2c(c1)CC2 c1(OC)oc(C)nc1C(=O)NCCCN(C(=O)CC1CCCC2CC12)C(C)C C(C(=O)NC1(C(=O)N(C)CCN(C2CC2)CC2CC2)CC1)=CCC C1(CC=C)(N(C(C2CC(CC)=NO2)=O)CC)CCN(C(=O)CCc2n[nH]c(=N)s2)C1 c1(COC(C2CN(C(=O)OC(C)(C)C)C3CCN2C3)=O)cc(F)c2ncccc2c1 c1(C(=O)OC)ccccc1C(=O)NC(C)CC(C)NC(c1coc(C(C)(C)C)n1)=O c1(C(N2CCN(C(CCC(C)SC)=O)CC(O)C2)=O)ccc([N+](=O)[O-])cc1C c1(C(=O)NC(CC(C)NC(=O)C(C)(C)CO)C)n[nH]c2c1NCCC2 CC1CN(C(c2cncc(O)c2Cl)=O)CCC1NC(C1(C(C)(F)F)CC1)=O c1(NC(C2C3CN(C(CC(=O)OC)=O)CC32)=O)cccc2cncc(F)c12 CCC1=C(C(=O)NCC2CCCN2C(c2cc3c(C)cccn3c2)=O)CCCO1 C1(CNC(C(=O)OC)CC2COC(C)(C)O2)COC2(CCC2)C1 c1(N2CC(N(C(c3c(CC)occ3)=O)C)C2)nc(Cl)nc2c(C(=O)OC)snc12 C1(C(N2CC(C(C)(C)NC(=O)CC3CCOCC3)C2)=O)C2CCCOC12 N1(C(C2(F)CCN(C(COC3(C)CCC3)=O)C2)=O)CCOCCC1C1CC1 C=C(C)C(CC(=O)N1CCC(CN(C(C2(CC(F)F)CC2)=O)C2CC2)C1)OCC c1(OC)ccc(O)cc1NC(=O)CN(C(C1CCCOC1C)=O)C(C)C N1(C(=O)Cn2cnnn2)CCC2(CC1)CC(Nc1ncc3ncnc-3[nH]1)CO2 N(C(=NCC1CCCC1)NCSC)CC(c1ncn(C)n1)O.C1(C)(CO)CCCCC1 C1(NC(c2cc(OC)ns2)C)CN(C)CC1C(F)(F)F c1(OC)ncccc1C(=O)NC(C)CCN(C)C(C1C2CCC1CC2)=O Cc1c(C(=O)NC(C(=O)NC(c2ccn(C)n2)C)c2ccoc2)cccc1O c1(C(N2CCC(=CCNC(C3C(C)C3)=O)CC2)=O)cc2cccnc2o1 N1(C(C(CCC)CC)=O)CC2CCCC(C1)N2C(=O)C(C)(C)C CCC(CNC(=O)C(N1CCC(Cc2noc(CC(C)C)n2)CC1)=O)(CC)CC c1(CCC(=O)N(C)CC2CCN(C(C(C)C3CCC3)=O)C2)cccnc1F n1(CC(=O)N(CCC)CCNC(c2ccc(O)nn2)=O)cnc2c1CCCC2 c1(C(=O)NCC2(F)CCC(NC(c3c(C(C)C)occ3)=O)C2)c(Cl)cccc1Cl c1(C(N2CCC(N(C(CC=C)=O)C)CC2)=O)[nH]c(=N)ccc1C Cc1cc(C)c(C(=O)NC(C2(O)CCN(C(=O)C3=CCSC3)CC2)C)c(C)c1 c1(C(N2CC(OC)C(F)C2)C(=O)NC)cc(OC(F)F)ccc1C Cc1ccc(C(=O)NCC2CCC(NC(c3cccnn3)=O)C2)o1 NC(=O)CCCCC(=O)NC1CCCN(C(=O)C=CC(c2ccccc2)=O)C1 c1(CC(N2CC(F)(C(=O)NCCCCOC(C)C)C2)=O)ccc(Cl)cc1 CCC(CC)CC(=O)N1CCN(C(=O)CC(O)CN(C)Cc2nccn2CC)CC1 c1(CC)cc(Br)ccc1C(N1CCCC1CNC(c1ccnn1C(C)C)=O)=O C(=O)(CCC1=CCCCC1)NC(CNC(=O)C1=CCCSC1)C1CCC1 N1(C(C(c2cc(C)sc2)(F)F)=O)CC(NC(=O)COCCCF)C(SC)C1 C(=O)(CC1CC(=O)c2ccccc21)N(C(C#N)C1CC1)CC1CC1 C#CC1(O)CCN(C(=O)CC2(CNC(c3ccc(F)cn3)=O)CC2)CC1 c1(C(N2CCC(NC(CC(C=C)(C)C)=O)C(O)C2)=O)ccc(F)c(OC)c1F C1(NC(c2cc(C(=O)OC)ncc2)=O)CC2(C1)CC(NC(=O)C(C)C(C)(F)F)C2 N1(C(c2n(C(C)C)ncc2)=O)CCC(CNC(C2(C)CCCCO2)=O)C(F)(F)C1 C(CC(CC)C(=O)N(CC(=O)N(C1CCOCC1C)C)C1CC1)=CC c1(C(=O)NC2C(C(=O)OCC)CCCCC2)cc2n(n1)CCN(C(C)(C)C)C2 C(=O)(C(O)CCc1ccccc1)NCCNC(c1ncn(C(C)C)n1)=O c1(COC)cccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2(C(N)=O)CC2)c1 N1(C(C(C#C)(C)C)=O)CCC2(CC1)CN(C(C1CC3CCCCC3O1)=O)CCO2 N1(C(CCCc2nc(C)sc2)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1C c1(C(=O)NC(C(C)NC(c2cnc[nH]2)=O)C)cnccc1SC1CCCC1 N1(C(Cc2cn(CC)nn2)=O)CC(NC(c2c[nH]cc2Br)=O)CC(F)C1 N1(C(C(C)n2cncn2)=O)CCC2(NC(=O)CCc3ncccn3)CCCC12 c1(CNC(C2CC3CC3N2Cc2cccc(O)c2F)=O)cccc2ccccc12 C(=O)(C(CCN(C)C)NC(C1CC=CC(O)C1)=O)NCC(n1cccn1)C N1(C(C2(C)CC(F)(F)C2)=O)CC2(CO)CC1(C(=O)NCCc1cc[nH]n1)C2 C1(S(=O)(=O)N(C)C)(N(C(C2CC2C)C)CC2CCCC2)CCC1 c1(C(=O)NC(C)CCNC(C2CC3(CC3)C2)=O)cc(O)cc(F)c1F C#CCC(C(=O)N1CC2C(C(N3CCC3(C)CCO)=O)C2C1)C1CC1 N1(Cc2cc(OC)cc(Br)c2)CCc2[nH]nc(C(=O)NC3COC(=O)C3)c2C1 n1(C(C2CCCCO2)C)cc(C2CC2C(=O)NCC2CCS2(=O)=O)nn1 CCCCCCCCCCN(C)Cc1ccnc2cccnc12 c1(Nc2scc(C(c3nnc(C)o3)C)n2)ccc(F)c(F)c1 CC(C(=O)NCC(O)CN(C(=O)CCC1OCCO1)C)NC(=O)C1CC1 C1(NC(C=CC=CC)=O)CCC2(CCN(C(=O)Cc3nc(=N)[nH][nH]3)CC2)C1 N1(CC(=O)N(C(c2ccccn2)C)C)CCCN(c2nnc(C(F)F)o2)CC1 C1(CC(=O)NCC(=O)NC(C)C)COC(C)(C)O1 c1(NC(CSCCC)=O)ccc(NC(c2ccc(O)c(C)c2)=O)cc1C c1(CC)c(C(=O)NC2(COC)CN(C(c3cc(CC(C)C)c[nH]3)=O)C2)cnn1C c1(C(N2CC3CC3(C(=O)NC3CONC3=O)C2)=O)ccc(Cl)cc1I C1(c2nnc(C(=O)OCC)s2)CCCN(C(c2nnc(C)s2)=O)C1 O=[N+]([O-])c1cccc(S(=O)(=O)N2CC3C(Br)C3C2)c1 c1(C(=O)NC2CCN(C(C34CCC(F)(CC3)C4)=O)CC2O)ccc2c(c1)OCC2 C(=O)(CCC(=O)NCC1C(O)C(O)CN1C(=O)CC1CC(=O)NC1=O)NCCC Cc1cc(C(=O)NC2CC(F)CN(C(C3(CN(C)C)CC3)=O)C2)cnc1O CCCCCC(F)C(=O)NCC1(C(=O)N(C)Cc2cccnc2)CC12CCC2 N(C(=NCCC(C)=O)NC(c1ccccc1F)C)CC(CC)CC(F)(F)F N1(C(CN(C)C(C2CCN(CCF)CC2)=O)=O)CC2CC(N(C)C)C2C1 N1(C(C2CCC(C)C2)=O)CC2CCCC2(NC(c2ccc(CN=[N+]=[N-])o2)=O)C1 N1(C(CC(COC)C)=O)CC2CCC(NC(=O)COc3cccc(C)c3)CC2C1 c1(OC)cc(-c2cccc(CC(=O)NCCN3CCN(C)CC3)n2)ccc1[N+](=O)[O-] C(CC(=O)NC1(CO)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)C1)(C(C)C)OCC c1(CN2CC3CN(C(c4c(C)nccn4)=O)CC32)cccc2nc[nH]c12 C1(CNC(=O)CCC2CC2)CC(F)CN1C(=O)COCc1ccccc1 N12CC(CC1(C)C)Nc1ncc(s1)C2=O.c1(OC)cc(C(=O)OC)ncn1 Cn1cc2c(n1)CCN(c1cc(NC3CN=CN(c4ccccc4)C3)ncn1)C2 CC(C)(C)CCCC(=O)N1CC2CC1C2C(N1CC2CC1C(F)(F)C2)=O c1(CC(=O)N(C2CN(C(c3cnn(C)c3)=O)C2)C)nccn1C c1(OCCC)cc(OC)ccc1-c1ccccc1C(=O)Nc1cccc(F)c1 n1(CCOC)ncc(C(=O)NCCC(O)CNC(C2(COC)CCOC2)=O)c1C C1(OCCCN(C)C(c2coc(Br)n2)=O)CCN(C(=O)C(C)(C)c2cnsc2)CC1 c1(OC)ccc(C)c(-c2cn(-c3cc(OC(F)F)ccc3C)nn2)c1 C1(O)(C(=O)NCC(C)NC(=O)C(C)N(C)C)CC(CF)C1 CC(N=c1[nH]c(=N)[nH]c(=NCC2(N(C)C)CCC(F)(F)CC2)[nH]1)c1cscn1 C1(C2CN(C(C3CC3CF)=O)C2)(NC(=O)C2=C(Cl)CC2)CC1 N1(C(c2c(CC)noc2)=O)CCCC1(CNC(=O)COc1ccsn1)COC C(=O)(CC(CC)C(C)C)N1C(CCn2cc(C(CC)O)nn2)CCCC1 CC(C)(CS(=O)(=O)N1CCCC(Cc2ccncc2)C1)C(F)F C1(NC(c2ccc(C(CC)C)cc2)=O)CCSC12CN(C(C1(C)CC1Br)=O)C2 c1(C(=O)NC2CC(OCC(=O)Nc3cccnc3S)C2)cc2ccccn2c1 CC(C)C(O)CC(=O)N1C(C(=O)NCC2(n3ccnn3)CC2)CC2CC12 n1(CC(=O)NCCc2cn(CCCF)nn2)nc(C(F)F)cc1C1CC1 c1(NC)ccc(C(=O)NCc2c[nH]nc2C(N2CC(O)(C(F)(F)F)C2)=O)nc1 CC(C)C(O)CC(=O)NCCC1CCN(C(=O)CC(O)CN(C)C)CC1 N#Cc1cc(F)ccc1C(=O)NCCC1(O)CCN(C(C2CCCO2)=O)C1 N1(C(c2cc(CNC(c3c(C)cc(C)s3)=O)on2)=O)CC(C)C(C)C1C c1(C(=O)NC2(C)CCN(C(c3cn(CCCC)nn3)=O)C2)nnc(O)cc1O Cc1cc(Br)c(CN(C(c2ccnn2C(F)(F)F)C(=O)NCC2CCCO2)C)s1 C1(NC(C2CC(C#C)(O)C2)=O)C2CC3C(C2)C13C(N1CC(=O)NC(C)C1)=O C1(C(=O)NC2C(SC)CN(C(=O)CCC(C)CN(C)C)C2)CC2(C1)CC2(F)F c1(C(N(C2CCCN(C(C3C(C)C3)=O)C2)CC2CC2)=O)ccc(S(N)(=O)=O)s1 C1(C(=O)NCC2(COC)CN(C(c3cnc(N)cn3)=O)C2)CCC(C)(C)O1 C1(C(=O)NCCC2CCN(C(C3(C)CCN(C)C3)=O)C2)CN(S(=O)(=O)N(C)C)C1 N1(C(COc2cc(C)on2)=O)CCC(CNC(C23COC(CCO2)C3)=O)C1(C)C CCC(N=c1[nH]c(=NCc2coc(C)n2)[nH]c2ccsc12)c1ccccc1N N1(C(C2(CC)CC2)=O)CCCC(C2CCN(C(c3cnc(C)[nH]c3=N)=O)C2)C1 N1(C(CCOC(C)C)=O)CCCCC(NC(C2CCC(F)(F)CC2)=O)C1 N1(C(C=C(C)Cl)=O)CC(C)OC2(CCN(C(c3ccc(N)c(F)n3)=O)CC2)C1 C(CC)(C(=O)N1CCCC1CCC(=O)NC1(CC)CCC1)OCC N1(C(c2c(NC)nccc2)=O)CCC2(CC2C(=O)NCC(c2cnc[nH]2)C)C1 N1(C(CCOCC(C)C)=O)CCCCC12CC(NC(c1cnnn1C)=O)C2 N1(C(COCCCCC)=O)CCC(CCN(C(=O)CC2CCCCC2C)C)CC1 c1(C(N2CCC(OCCn3cc(Cl)cn3)C2)=O)cncc2c[nH]nc12 Cc1nn(CC(C)C)c(C)c1CC(N1CC(N(C)C(c2ccoc2)=O)C1)=O Cc1ccc(CC(=O)NCC23CC(NC(c4ncc[nH]c4=O)=O)(C2)C3)cc1O C=CC(C)C(C)C(=O)N(CCNC(c1ccc(C)c(NC(C)=O)c1)=O)CCSC C(C(N=[N+]=[N-])C(=O)NCC1(CO)CN(C(=O)Cc2cccc(OC)c2)C1)OCC c1(NCCCNC(C(c2cccs2)SC)=O)cc(C)nc2ncnn12 N1(C(c2cc(N)c(O)cc2)=O)CC2CCC1CCN2C(=O)C=CC1CCCC1 Cc1cc(C)c(CNC(C2CCOC2CNC(=O)Cc2cccnc2F)=O)cn1 N1(C(C(C(C)O)C)=O)CCC(C2(NC(c3cnc(O)c4ccsc34)=O)CC2)CC1 c1(C(=O)NCCNC(CNS(N(C)C)(=O)=O)=O)cc2cccc(Br)c2o1 C(CC(C(C)(C)C)NC(c1cnn(CCF)c1)=O)NC(CN(C(C(C)C)=O)C)=O c1(OC)ccc(Br)c(C(N2CCN(c3nc(C)ncc3Br)C3CC23)=O)c1F CC1=CCC(C(=O)N)CC1.C1(CC=O)CCN(C(=O)C(F)F)C1 C1(NC(c2oc(SCC)c(C)c2)=O)CCC2C3CCC(C3)C12 c1(-c2ccc(C)c(C)c2)ccc2c(c1)CCN(C(c1c(F)cc(I)cc1F)=O)C2 NC1(CO)CCN(C(=O)C(N2CCC(c3ccccn3)CC2)=O)C1 Nc1ccc2nc(N3CCOCC(NC(C4CC5CC5C4)=O)C3)sc2c1 CCCC(CCCNC(c1cc(C)n(C2CC2)c1C)=O)NC(=O)CC(F)F C1(NC(C(C=C=C)C)=O)CC2CC(C1)N(C(=O)CSc1nncs1)C2 C(CCCC(C)Sc1ccccc1)N(C(c1c(C)non1)=O)CC1(F)CCOC1 Cc1ccc(C(=O)NC(C(=O)NC(C)C(F)F)C2CCCC2)cn1 C12(NC(Cc3c(C)scc3)=O)CC3CCC(C1C2)N3C(C1CCCCC1(F)F)=O C(CCC(=O)NCc1csc(C(C)=O)c1)SC.C12CCN(C1)C2=O C1(NC(C=CC)=O)CCC(O)CN(C(C2CCN(C3CCC3)C2)=O)C1 N1(C(=O)O)CCCCC2(C1)CN(C(C)=O)C2.C(CC(C)C)(C(=O)NOC(C)(C)C)OC C(CC1CC1)(CC(=O)NCC(C)CCCO)NC(c1cc(C(C)=O)on1)=O c1(-c2ccc(OCC)nc2)nc(C(=O)Nc2cccc(F)c2I)n2ccccc12 N1(C(C(C)OCCCC)=O)CCC2(CC1)CC2C(N1CCn2nccc2C1)=O C#Cc1ccc(CNC(C2(C(C)NC(C3CC4CCCC4C3)=O)CC2)=O)cc1 N1(CC)CC2(CCOCC2)C1c1ccn(CSCc2ccccc2[N+](=O)[O-])n1 Cc1cc(NC(C2CCN(C(=O)C(O)C(C)(C)C)C23CCC3)=O)cc(C)c1F C(C(CC(=O)NCCCCCNC(C1(C(F)F)CCC1)=O)CC(C)C)NC(C)=O C1(NC(C2CC(C)(C)O2)=O)CC(F)CN(C(c2csc(Cl)n2)=O)C1 N1(C(c2cc(C)oc2C)=O)CCN(C(C2CCSCC2)=O)C2CCCCC12 c1(C(=O)NC2C(CNC(=O)CSC(F)F)CCC2)ccc([N+](=O)[O-])s1 CCCCCC(C)CC(=O)N(CC(O)CN(C)C(c1cnc(C)cc1C)=O)C c1(NC(N2C(C3(O)CN(C(c4c(C)nsc4)=O)C3)CCC2)=O)occ2c1CCC2 Cc1cc(CC(=O)NC2CC(F)(CNC(C3COC(=O)C3)=O)C2)cc(C)c1 c1(C(=O)NC(CC)CNC(=O)C(C2CCCC2)SC)ccc(OC(C)C)cc1 N1(NC(C=CC)=O)CC2(C)CC1CCO2.c1(C)ccc(C(F)(F)F)cc1C C(C1CCCN1C)=CC(N1C(C2(NC(COCCC#C)=O)CC2)CCC1)=O C(=O)(CCCC1CCC1)NCCN(CCOC)C(c1csnc1Cl)=O C(=O)(CC1=CCCC1)NC(C1CN(C(c2cc(F)c[nH]2)=O)CCO1)C CN1CCC(CCN(C=O)CC2CN(C(=O)OC(C)(C)C)CCCO2)OC1=O CC1(C(N2CC=CC(NC(=O)CSc3nncn3C3CC3)C2)=O)CC(=O)CCO1 N1(C(CSc2ccc(OCC)cc2)=O)CC2(C1)CN(C(=O)C(CO)OC)CCO2 C(=O)(C(C)=Cn1ccnn1)N(CC(N1CCN(C(C(CCC)(C)O)=O)CC1)=O)C N1(C(C2C(CNC(C3C(C)SCCC3)=O)CCO2)=O)CCC(C)(O)C(O)C1 C1(C(=O)NC2CC2)CCN(C(C2CC(OC)C2)=O)C12CCC2.c1(OC)ccnc(S)c1 C(=O)(C1=C(C)CCC1)NCc1[nH]nc(C2CCN(C(CCCC#C)=O)CC2)n1 CN1CCCCC1C(=O)NCC=CCC(=O)NCCC(O)C1CC1 C1(CC)(CC)CCCN(C(=O)CCCNC(=O)CCc2cn[nH]c2)C1 N1(C(N2CCCN(Cc3ccco3)CC2)=O)CCc2c(ccnc2Cl)C1 C(C(CCO)NC(=O)C(c1ccoc1)NC(C1CC(C)(O)C1)=O)OC N1(C(c2ccc(OC)s2)=O)CCC2C(CCCN2C(c2ocnc2C(F)F)=O)C1 c1(C(=O)NCC(C)(CNC(C2CCCC2O)=O)OC)ccccc1CO c1(C(=O)NC(C2(CNC(c3nc(CC)oc3)=O)CC2)C)cc(OC)ccn1 N1(c2sc(C(=O)OCC)c(C)n2)CCC(O)(CN)CC1 C1(C(N(C2CCN(C)C2=O)C)=O)CCCN(C(c2ccc(Cl)cc2)=O)CC1 C1(c2ccc(C)nc2Br)NC(=O)N(CC2CCCCC2)C=NC1(C)C C(=O)(C1CCCc2cncn21)NC1CN(C(c2c(C(C)C)[nH]cc2)=O)CC1(C)C c1(C(=O)NC2CCC(CNC(c3c(C)nc(N)cn3)=O)C2)cc(F)c(F)cc1F c1(CC)cc(C(=O)NCC23CC(NC(c4cnccn4)=O)(C2)C3)cc(O)n1 c1(OC)ccnc(C(=O)NCC(C)(CC(C)C)NC(c2cn(C)nn2)=O)c1OC CC(C)C(C(=O)N1CCCc2c(Br)cnn21)C(C)C C1(CC)CCN(C(=O)Cc2nocc2C)C1C(N1CC[Si](C)(C)C1)=O C12(C(N3CC(OCc4cn(C(CC=C)CC=C)nn4)C3)=O)CCCN(CCC1)C2 C1(C(=O)NC(C(=O)NC(C#C)C(C)(C)C)(C)CSC)CC2CC(=O)C1O2 N1(C(CCC2N(C)CCC2)=O)CCC(C2(NC(=O)Cc3cccs3)CC2)C1 c1(NC(CCCC=C)c2nnnn2CCCSCC)csc(S(N)(=O)=O)c1 Cc1nc2c([nH]1)CC(C(=O)NCC(C)(CC(C)C)NC(=O)CN(C)C)CC2 c1(CC(C)C)ccc(C=CC(N2CCCC(NC(C3(C)CC4CC4C3)=O)C2)=O)cc1 C1(NC(C=C(C)C2CC2)=O)CN(C(=O)C#CC2(C)CCCO2)C2CCCCC12 C1(n2cc(C34OCC(CNC(CCCC(N)=O)=O)(C3)C4)nn2)CCCCC12CC2 C12(C(=O)NCCN(C(=O)C#CC3CC3)CCCCCC)CCN(CC1)S(=O)(=O)C2 N1(C(=O)CCN(CCO)CCO)CCOCC1C1CCCC1 C12(CNC(CC(=O)OCC)=O)CCC(CNC(c3ccc(C)c(C)n3)=O)(CC1)OC2 c1(C(=O)NCC(C)N(C)C(C2CC(=O)N(C)C2)=O)cc(F)ccc1Cl CCC1=C(C(=O)NC2CC2CNC(=O)Cc2csc(C)n2)SCCO1 CC(CO)CCCNC(=O)C(C(=O)OC(C)(C)C)NC(=O)C(C)(O)C1CCC1 C1(C)(C(=O)NCC(CC)NC(=O)CCC2CCCN(C)C2)CC(=O)N(C)C1 c1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)N(C)C)C2)cc2nc(Cl)ccc2o1 c1(C=O)cc2cccnc2o1.N12CCC(C1)SCCC2=O.c1(C(=O)N)cnc(O)o1 CCC(CNC(c1cccc(C)n1)=O)(CC)NC(=O)CC(C)CN(C)C C(=O)(CCC(=O)NCC1CC(NC(=O)COC2CCC2)C1(C)C)N(C)C C1(C(=O)NCc2c(C(=O)NCCc3ccc(C)s3)occ2)CCC(F)(F)C1 N1(C(CCN(CCC)C)=O)CC(=O)CC1C(=O)NCC(C)(C)C1CCCO1 C1(NC(C(C)c2ccco2)=O)CN(C(c2cc(O)nc(Cl)c2)=O)CC1(C)C C(=O)(C(Cc1ccccc1)NS(C)(=O)=O)NC(C)CCNC(C1CC1F)=O c1(C(=O)NCC(CC=C)NC(c2n[nH]cc2C2CC2)=O)nn(C)c(=O)cc1C c1(SC)ccccc1C(N1CCC1CNC(C1(C)COCCO1)=O)=O C=C=C(C)CC(=O)NC1CN(C(C23CSCC2C3)=O)CC1C(F)F CC1(C)CCN(C(C2CN3CCC2CC3)=O)C(C(=O)NC2CNC(=O)OC2)C1 CC1CC2(CCN(C(=O)CC3NC(=O)NC3=O)CC2)CN1C(=O)C(Cl)=CCl Cc1cnc2ccc(C(=O)N(CC(O)CN(C(=O)Cc3ccoc3C)C)C)cn12 C=Cn1nccc1C(=O)NC(C1CCCC1)CNC(C1CC(N=[N+]=[N-])C1)=O c1(NS(=O)(=O)CC2CCCCNC2)cnc(C2CC2)cn1 Cc1cccc(S(C)(=O)=O)c1-n1cc(S(=O)(=O)NCCCC2CCCCC2)nn1 Cc1nc(-c2ccccc2Br)sc1CCN(C1CC2CC1CN2)C(C1CC(=O)N1)=O c1(C(N(CCCNC(=O)CNC(c2cscn2)=O)C)=O)cnc(N)c([N+](=O)[O-])c1 N1(C(C(CC)CN(C)C)=O)Cc2n[nH]cc2C1C(=O)Nc1ccc(O)cc1C c1(OCC2(CNC(=O)NCC3C4CCCOC34)CC2(F)F)ccc(F)cc1F c1(CCC2CN(C(N3CCN(C(=O)OC(C)(C)C)CC3)=O)C2)cccc(F)c1N c1(CC)oc(C)cc1C(N1CC2C(NC(=O)CCc3ncc(C)[nH]3)C2C1)=O C1(C(N(CCCCNC(c2cc(F)cs2)=O)C)=O)CC2(CC2)CN1C N1(C(C(=Cc2cccnc2)C)=O)CCC2CN(C(C3CCC3(F)F)=O)CC12 N1(C(c2cccnc2Nc2cccnc2)=O)CCC2(CC1)OCC1CC21 C(c1cccc(O)c1)=CC(N1CCCC(CC(=O)NCCC2N(C)CCC2)C1)=O C1(c2n(C)ncc2)OCCC1N=c1[nH]nc(C2CC2)s1 c1(NCc2cn(CC3N(C(C(CC(C)C)O)=O)CCC3)nn2)ccc2[nH]ccc2n1 C1(CC)(NC(=O)C=NOC)CCCN(C(C2CCCCNC2=O)=O)C1 C(=O)(CCCCCC#N)N(CCC(=O)NC(c1cccnc1O)C)C(C)C C1(NC(C(CC2CC2)OC)=O)CC2CC1N(C(c1n[nH]cc1F)=O)C2 C(=O)(CCCCCC)NC1C(CNC(C(C)OCC=C)=O)C1 c1(OC)c(Cl)ccc(C(N2CCC(NC(=O)C(F)(F)c3cscn3)C2)=O)c1N c1(C(N2CCC(F)(CNC(C3CC3(Cl)Cl)=O)CC2)=O)c(O)ccc(F)c1F C1(CC=C)(N(C(=O)C(CC)CC)CC)CCN(C(=O)C(C(C)C)C2CCC2)C1 c1(C(N(C2CC3CC(C2)N(C(=O)C2CC2)C3)C)=O)ccc2c(c1)CCCC2(C)C C1(C(N(C(C)CC(F)(F)F)C)=O)N(C(=O)OC(C)(C)C)CCC1(C)C Cc1ccc2c(c1)SC(C(N1CCC(C3(NC(c4ncn(C)n4)=O)CC3)C1)=O)C2 O=S(=O)(c1cccc(=NC2CCC(CCO)CCC2)[nH]1)NC1(CO)CC=CC1 C1(OCC)CC2CN(C(C3CC(C)N(C(=O)C(F)C(C)C)CC3C)=O)CC12 C(CCNC(=O)CCc1ccc(F)cc1)(C(C)C)NC(c1cn(CCC)nc1)=O CCCC(CC)NC(=O)NC(C(=O)OCC)C1CCC1 CC1CC(NC(=O)C(C(C)(C)C)NC(N)=O)CCN1C(=O)Cc1nccn1C CC1(C)CC(CO)CN1C(c1cccc(Cc2cn(CC3CCCCN3)nn2)c1)=O Cc1cc(C#N)ccc1-c1cn(C(N2CCCC(C)(C)C2C)=O)nn1.c1(C)ncon1 CC1CCCCC1C(=O)NC1CCN(C(c2cc(C3CC3)[nH]n2)=O)C1C C=C(C)CCCCNC(=O)C(C1CCOC1)NC(c1[nH]nnc1CC#N)=O c1(C(=O)NC(CNC(CC(C=C)C)=O)C)cc(S(N)(=O)=O)ccc1Br C1(C(=O)OC)CC2(CC(NC(=O)NC(c3cccc(F)c3OC)C(F)(F)F)C2)C1 c1(C(N(CCCCNC(C(C2CCOC2)OC)=O)C)=O)cnc(CC2CC2)nc1O N1(C(c2c(CCC)n(C)nc2)=O)CCN(C(C2COCC(C)O2)=O)C2(CC2)C1 CCCCC(C)C(=O)N(C(C)CN(C)C(c1ccccc1-n1nccn1)=O)C C12(NC(C(CC#C)CC#C)=O)CCCC1(F)CN(C(C1(C3CC3)CC1)=O)C2 O=C(CS(=O)CCC(F)(F)F)NC1(CF)CCN(C(c2ccnn2C(F)F)=O)C1 c1(CC)cc(CCC(=O)NC(C)(CNC(=O)C(C)(C)OC(CC)=O)CSC)oc1C CC1(C)CC(C(=O)N2CCC(CN=c3[nH]nc(COC)s3)C2)=NO1 c1(C(c2cccc(N)c2)NC(=O)NC2CCC(n3cccn3)CC2)ccc(F)c(Br)c1 C12(OC)CCCCC(C(=O)NC3(CNC(C4COC(=O)N4)=O)CCOC3)(C1)C2 c1(C(=O)NCCCN(C)C(C2CCCN2C(c2ccsc2)=O)=O)ccc(O)cn1 c1(C(N2CC=CC(NC(CN(C3CCSC3)C)=O)C2)=O)cc2c(nn1)CCCC2 C(=O)(CC(C)CC(=O)NCC1(C)CCC(NC(c2cnc(C)o2)=O)CC1)OC Cc1noc(C)c1C(C)C(=O)NCc1ccccc1NCC1CCCCO1 C1(CCNC(c2cnn(CC)c2Cl)=O)C(C)CCCN1C(=O)COCCF C1(C(=O)NCCN(C(c2cnc(COC)[nH]2)=O)CC)CCCN1S(C)(=O)=O C1(NC(CC2(C)CC2(F)F)=O)CC(NC(=O)COc2cccnc2)C12CCC2 c1(C(=O)NCC(C)CNC(=O)CCC2CCCCO2)cccc2c[nH]nc12 N1(C(CC(C)C(C)(C)NC(C2CCCO2)=O)=O)CCC2(CNC(=O)N2)C1 C1(NC(=O)CSCc2ccccn2)CCCN(C(=O)Cn2ncnn2)CC1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1C(CNC(=O)CSc2ccccn2)CC1 C#CCCCC(C)C(=O)NC1CC(C)(NC(=O)CCCc2ccc(O)cc2)C1 C(=O)(C(F)CC(C)(C)NC(=O)CC1(C)CCOC1)NCC1(OC)CC1 C1(Nc2c(C(=O)OC)ccc(C(F)(F)F)n2)CN(C(C)=O)C2(CCCC2)C1 c1(OCC)ccc(Cl)cc1CC(C)(C)NCC(C)(O)C(C)(C)O c1(OC)c(C(=O)NC2CCCC2NC(=O)CS(=O)(=O)N(C)C)csc1Cl C1(C(=O)NCc2ccc(CNC(=O)CC3C=CCOC3)cc2)CCC2(CCC2)C1 c1(NC(CN(C)CC)=O)cc(OC)c(OC)cc1Br.C1C(C(C)C)NC(=O)N1 C1(CCC)CN(C(=O)C(CC)SC)CC1C(=O)NCc1cccc(C)n1 CC1CC(CNC(C2CCNC(=O)C2)=O)CCN1C(=O)CCC1(C)CC1 Cc1cc(C(=O)NNC(=O)N(CCCO)C(C)C)cc([N+](=O)[O-])c1Cl c1(CC(N2C(CNC(c3cnncc3O)=O)CCCC2)=O)ccc2n[nH]cc2c1 C1(NC(C(CCOC)C)=O)CC(F)(F)CC1NC(c1sc(C)cc1C)=O C1(C(N(CCN(C(C23CCCCC2C3)=O)CC)CC)=O)C2CCC3C(C2)CC13 Cc1ccnc2c(C(N3CC(CNC(c4ccnnc4)=O)CC3(C)C)=O)cnn12 CC1(CCNC(C2CCS(=O)(=O)C2)=O)CCN(C(c2coc(C(F)(F)F)n2)=O)C1 C(N=c1[nH]c(Cl)nc(C)c1F)C1C(C)CCN(C(CCn2ncc(C)c2)=O)C1 c1(C(=O)NC)ccc(C(N2CCCC2CNC(=O)C=Cc2cn[nH]c2)=O)cc1F c1(CNC(=O)NCC2CC3OCCC3O2)c(F)cc(Cl)cc1F C1(S(C)(=O)=O)(C(=O)NCC(CNC(Cc2c(C)n(C)nc2)=O)C)CC(O)C1 Cc1noc(N)c1C(=O)NC1CCC1NC(c1cnn(C(F)F)c1)=O c1(CC)noc(CCC(N2CCCC2CN(C(=O)C=CI)CC)=O)n1 C1(CNC(CSCCN(C)C)=O)(NC(C2CCCO2)=O)CCOCC1 c1(C(=O)NCC2CN(C(c3scc(OC)c3)=O)C(C)CC2)ccc(F)c(C#N)c1 C#CC(C)(C)C(=O)N(C1CC(NC(c2nccnc2C)=O)C1)C C1(C(=O)NCC2CC(NC(C3(CC4CCC4)CC3)=O)C2)C2CCC1CC2 C1(C(=O)NC2C3(CC(NC(Cc4cc(OC)no4)=O)C3)C2)CCC([N+](=O)[O-])CC1 C1(CC)CN(C(C2CN(CC(F)(F)F)C2)=O)CCC1NC(c1cc[nH]c(=N)c1)=O C1(C(=O)NCCc2c(C)nccn2)CC2C=CC1N(C(c1ccsn1)=O)C2 C#Cc1cccc(C(=O)NC2(CNC(c3cncnc3C)=O)CC2)c1F CN1CCOCC1(c1cn(CC(N2CCC(CN(C)C)C2)=O)nn1)CO C1(CNC(C2CC(CC3CC3)C2)=O)CN(C(C2(C3CCC3)CC2)=O)C2(CCC2)C1 C(=O)(C1=CC2CCC(C1)C2)N1CC(NC(C=COCC)=O)(COC)C1 N1(CC(=O)NCC(CC(F)(F)F)NC(c2ccc(O)nc2)=O)C(=O)CCCC1=O c1(N2C(C)(C(=O)NC3CC(CSC)C(O)C3O)CCC2)ccc(Br)cc1[N+](=O)[O-] N1(C(C(CCC)NC(N)=O)=O)C2CCC1CN(C(C1CC1(C)CC)=O)CC2 C1(CCC)(C(N2CC(Cn3cc(CNS(=O)(=O)C(C)C)nn3)C2)=O)CCNC1=O C1(NC(C(C)(CO)OC)=O)CC2CC1CN2C(c1cccnc1)=O N(C1CS(=O)(=O)c2ccccc21)CC(CC)C#N C1(N(C(CC2(CC(C)C)CC2)=O)C)CCC(CNC(C2CCN(C)C2C)=O)CC1 N1(Cc2c(C(C)(F)F)n[nH]c2)CCCC(N2CCCCC2)C1 c1(C(=O)NCC2C3CN(C(CC)=O)CC32)ccc(=NC)[nH]c1 C(=O)(C(F)C(C)C(F)(F)F)N1CCN(C(Cc2ccc(SC)cc2)=O)C(C)C1 C1(C(=O)NC2C(CNc3nccc(C(=O)OC)n3)CCC2)CC2(CCCC2)CO1 C1(CN2CCCC2)CCC=CCCC1.N12CCN(CC1)C(=O)c1ccc(o1)C2=O C(CC1CCCO1)(C(=O)NCCCCC1CCCC1)NC(=O)CCc1cscn1 c1(C(=O)Nc2cc(C)sc2)cccc(CNC(=O)CCc2c(C)noc2Cl)c1 C1(C(=O)NCCOCCN(C(=O)C(F)CC2CC2)C)C2CC3CC(C2)CC1C3 CCC(=O)CCC(=O)N1CC2(CC2)CC1C(N1CCC2C(C(N)=O)C2C1)=O Cc1cc(=NC(C)C2CCCN(C(c3cn4cc(Cl)cnc4n3)=O)C2)[nH]c(C)n1 N1(C(CCCOC(C)=O)=O)CCC2(CCN(C(=O)CC3C(=O)NN=C3C)CC2)C1 c1(C(=O)N(C(C2(O)CN(C(C(C)C)=O)C2)C)C2CC2)nc(C2CC2)cs1 N1(C(c2c(CC)n(C)nc2)=O)CC(NC(=O)C(C)OCC(C)C)CC1(CC)CC C1(CNC(c2c(C)nc(O)[nH]2)=O)CCN(C(=O)Cn2cnc(C#N)n2)CC1(F)F Cc1nc(C(C)C)oc1C(=O)NCCCNC(C1CC=CCC1)=O N1(CC(=O)NCC2CCN(C(c3ccc(C)[nH]3)=O)C2)OC(C)(C)CC1=O n1(CC)cccc(NC(=O)C(C)(C)CNC(=O)C=Cc2cscn2)c1=O c1(C(COC)NC(=O)C(C2CCCOC2)NC(=O)OC(C)(C)C)ncccn1 N1(C(CNC(CC)=O)=O)CCC(C)C(CNC(C2CCCCN2C(N)=O)=O)C1 c1(C(=O)NCCCN(C(c2cccc(CC)n2)=O)CC)cccc2cncn12 N1(C(c2ccc(N(C)C)cc2)=O)CC2CC(C1)CN(C(c1cncs1)=O)C2 C(C)(C(=O)N(CC(CO)NC(=O)NCCOC)CC)NC(C)=O CCC(COC)C(=O)N(C1CCCCC1NC(c1cnc(-c2ccco2)s1)=O)C c1(C(=O)NCCCNC(CC(C)C(F)F)=O)c(O)ncc2c1CCC2 CC1CN(C(c2cnn[nH]2)=O)CC1CNC(=O)C(O)Cc1cccc(Cl)c1 C(CC(C)C(=O)NC1CN(C(=O)Cc2cnns2)CC1OC)=CCC c1(C(N(CCN)C)=O)ccc(NC(=O)C(C)=O)cc1.C1(C(=O)NC)CC2CC2C1 O=C(C(O)C(F)F)NCCSc1ccc(-c2cn(-c3cccnc3)nn2)cc1 N1(C(=O)Nc2ccc(NCc3ccccc3)cc2)CCN2CC(O)CC2C1 c1(N2C3CN(C(C4C(C)CCCC4)=O)CC2CC3)nc(Cl)nc2cnn(C)c12 C#CCCC(C(=O)O)NC(=O)C(C)Oc1ccccc1Br C12CCC(CC1)C(=O)N2.N1(Cc2scc(C)n2)CCS(=O)CC1 c1(C(N(CCOC)C2CC2)=O)cc(=O)n(C)cn1.C1(=O)C(F)C=CCN1 c1(OC)ccc(Br)cc1CC(N1CC2CC2(C(N2C(C(N)=O)CCC2C)=O)C1)=O c1(C(N2C3CCC2CC3)=O)ncc(N2CCOCC2)c(N2CCOCC2)n1 C(C(CN=c1cccc(S(=O)(=O)NC(C)CN2CCCCC2)[nH]1)C(C)C)OC C1(NC(=O)CCC2CCCCCC2)CN(C(=O)C=C2CCC2)CC12CCC2 CC1CCCC(C(=O)NCC(C)=CC(=O)NC2(C3CC3)CC2)CC1 N1(C(C(C(=O)OC)OC)=O)CCOC2(CCN(C(=O)C(C)(C)C3CC3)CC2)C1 C1(C(N(C2CCN(C(c3cnn(C4CC4)c3)=O)C2)CC)=O)CC2(CCO1)CC2 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(C2CC(=O)N2)=O)CC2(C1)CCC2 C(CC(C(=O)NC(C)(C)CC)NC(=O)CN1CC(C)(OC)C1)=CC Cn1cncc1C=CC(N1CCCC(CCNC(C2CC2c2ccsc2)=O)C1)=O N1(C(Cc2c(OC)cccc2)=O)CC2CCC1CN2C(c1cc(=O)cc(Cl)[nH]1)=O C1(C(N2CC3N(C(C4C(CCOC)C4)=O)C(C3)C2)=O)CC2CCCC(C1)C2 C1(C(=O)NCC(C)=CC(=O)NC(c2ccccc2)CO)CCN(C)C(=O)C1 c1(C(=O)NCCC(C)N(C(CSCC)=O)C)[nH]c(C)c(C(F)(F)F)c1C CC1(C)COCC(CC(=O)NC2(C)CCN(C(=O)Cc3cscn3)C2)O1 c1(C(C)NCC=CCNC(C=COCC)=O)ccc(C)cc1 c1(Cc2nc(C(CCC)C)nn2-c2cnn(C)c2)cc(C)cc(F)c1 N1(C(C(=Cc2ccc(F)cc2)C#N)=O)CCC2CN(C(=O)C3=CCC3)CCC2C1 CC(CNC(=O)C(C)(C)c1cccs1)CC(=O)NC1(O)CC2CC1C2 C(CC(C(=O)N1CCCC(C(C)C)C1)NC(=O)COC1CC1)=CC N#Cc1cccc2c(CN3CCN(Cc4ccc5ccccc5c4)CC3)c[nH]c12 c1(C(=O)NCC(CN(C(CCCC(=O)OC)=O)C)C)cc2nnn(C)c2s1 C(CC1=CCN(C(=O)Cc2cc(F)cc(F)c2)CC1)NC(c1cc(C)c(Cl)s1)=O C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(C(C)=C(CC)C)=O)CC=C1 C1(NC(CN(S(C)(=O)=O)C)=O)CCC(NC(=O)C(F)n2cccn2)CC1 c1(C(=O)NCC2CN(C(C(CCSC)(C)C)=O)C2)cc2cc(C)ccc2o1 N1(C(CC(CC)C2CC2)=O)CC(CC(=O)NCC=C2CCOCC2)C2(CC2)C1 CC(C)C(O)C(=O)NC(CNC(=O)C(C)C1CCCO1)C(C)(C)C C(C1CC(=O)N(C)CCO1)NC(COC(C(=O)OC)C)=O.C(COC)OC C1(C(C(=O)NCC(=C)C)N(C2CC2(C)C)CC)CC12CCC(F)(F)CC2 Cc1nnc2n1CCC2(C)C(=O)NCC(C)(C)CNC(=O)C(C)S(N)(=O)=O Cc1ccc(Cl)c2sc(NC(=O)C(N3CCC(C)C4CCCCC34)=O)nc12 N1(C(=O)NC2C(c3cccc(C)c3)CCCC2)CCC(C(=O)N(C)C)C12CCCC2 C1(NC(Cc2c(C)ccs2)=O)CN(C(=O)Cc2cncc(O)c2)CC(C)(C)C1 C1(CNC(C(c2n(C)ncc2)(F)F)=O)CC2COCC2N1C(=O)CCS(N)(=O)=O C1(C(=O)NCC2(NC(c3ccccc3)=O)CCCC2)CCCN(CC(F)(F)F)C1 c1(OC)cc(C)c(C(N2CC(NC(c3ccccc3O)=O)C(F)(F)C2)=O)cn1 C1(C(F)(F)F)(C(N(C2CCCN(C(C3COCCOC3)=O)C2)C)=O)CCOCC1 Cc1oc(Br)cc1C(=O)NCCC(C)CCNC(c1nn[nH]c1Cl)=O c1(-n2ccc(C(N)=O)n2)nc(-c2ccccc2-c2ccco2)cc(O)n1 N1(C(c2ncc(NC(C)C)nc2)=O)CC(C)CCC1CNC(=O)Cc1ccsc1 C1(C2CCN(C(=O)CCC(C)(C)F)C2)(NC(C2N(C(C)=O)CCC2)=O)CC1 c1(C(N(CCNC(c2ncsc2C(C)C)=O)CC)=O)ncnn2cccc12 c1(NCC2CCC(NC(=O)OC(C)(C)C)OC2)coc2c1C(=O)NCC2 CC(CCC(=O)NCC(CNC(c1ccnn1C(C)(C)C)=O)CO)N(C)C C(CN=c1nc(CC)cc(C)[nH]1)C1CCCC(NC(C=COCC)=O)C1 CN1CCN(C(=O)CN2CCCC2)C(C(=O)NCc2cc(O)ns2)C1 C1(C#N)(C(N(C2CCN(C(C(CC)OCC)=O)C2)CCO)=O)CCCC1 CC1CCN(C(=O)C=CC2CC2)CCN1C(=O)OC(C)(C)C c1(C(=O)NCCCC(=O)N(CC(O)CNC(=O)CSC2CC2)C)ccc(O)cc1 C12(CNC(C(C)(C)C3CC3)=O)CCC1CCN2C(c1cncc(C2CC2)c1)=O c1(C(N2CCC(C(N(CC(C)C)CCC)=O)CC2)=O)cnn2ccccc12 S(=O)(=O)(c1ccc2c(c1)CC(C)(C)O2)N1CCN(CC(C)CO)CC1 C1(CC(C)C)CCN(C(=O)CN(C(=O)C(c2ccccc2)O)C)C1 Cc1cnc2nc(-c3cccc(C(=O)N=S(C)(=O)C4CC4CO)c3)sc2n1 N1(C(C2CN(C(C(COC)COC)=O)CC2C(N)=O)=O)CC2(C)CC1(COC)C2 C=CC(CC)C(=O)NCC1COCC1NC(C1(N(C)C)CC1)=O c1(C(=O)OCc2c(C)nn[nH]2)cccc2nnn(C)c12 CC1Cc2cc(C(=O)N(C)CCN(C(=O)CC3CCC(O)CC3)C)ccc2O1 C1(CC=C)(NC(=O)C(c2ccccc2)C)CCN(C(c2cc(C)c(C)s2)=O)CC1 C1(C(N(C(CNC(Cn2ncc(CC)c2)=O)C)C)=O)CC2(C1)CC(C)(C)C2 N1(C(C=CCC)=O)CCc2nc[nH]c2C12CCN(C(C1CNC(=O)CC1C)=O)C2 N1(C(CCC2CCN(C(C3N(C(C)=O)CCC3)=O)C2)=O)CC(O)C(O)C1 c1(C(N2CCOCC(CNC(C3C(C)(C)C3)=O)C2)=O)cc2c(O)ncnc2cn1 c1(C(=O)NCCC(C)NC(C2CCC(C(=O)N(C)C)C2)=O)cnn2cccc2c1 CC(C(=O)N1CC2CC(NC(=O)Cc3csc(Br)n3)C1C2)C(C)(C)O Cc1cnc2nc(C(N3CCC(N(C(=O)CC4CC=CC4)C)C3)=O)nn2c1 C1(CNC(C2(C)CC=CCC2)=O)CN(C(=O)C(F)=C2CCC2)CC12CC2 Cc1ccc(C(=O)NCC(CNC2CCCC2)C(F)(F)F)cc1[N+](=O)[O-] CC1CN(C(C2(C(N)=O)CC2)=O)CC1CCNC(=O)CC1(C2CCCC2)CC1 c1(C(C(=O)NC)N(C(C)CC(C)C)C2CC2)cc(OC)ccc1F CCC(C(=O)NCCSCC(=O)Nc1cc(C)ccc1F)C(C)C C1(NC(C=C(CC)CC)=O)C2COCC1CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 C12(C(=O)NCC3ON=C(C(=O)N(C4CC4(C)C)C)C3)C(=O)C3CC1C2C3 C1(N(C(C=CC(C)C)=O)C)CCCC(NC(C(=O)N(CC(F)(F)F)CC2CC2)=O)C1 C1(NC(C2ON=C(C(C)C)C2)=O)CCC2(CC1)CCN(C(=O)C=CCF)C2 Cc1c(Br)c(C(N2CCCCC2C(C)NC(C2(F)CC=CC2)=O)=O)nn1C C1(C)(C(N2C(CCC=C)CCC2)=O)CC(O)CN1C(=O)CC1CC1COCC N1(C(C(C(=O)OC(C)(C)C)OC)=O)CCCC(CNC(=O)C2=COCCO2)CC1 S(=O)(=O)(c1ccc(F)c(Br)c1)N1CC2CN(C(=O)Nc3cc(C)cc(C)c3)CC21 N1(C(c2c(OC)ccs2)=O)CC(C(=O)N(C(C)C(C)(C)C)C)C2(CC2)C1 C1(C(=O)NC2CC(CNC(C=CC(=O)N(C)C)=O)C2)CS(=O)(=O)CC12CC2 C1(C(=O)NC(CCC=C)C)CC(O)CN1C(=O)CN1CCCCC1C N1(C(c2c(C)cc(C(F)F)o2)=O)CC2CCC(C1)N2C(=O)CCC1CCOC1 c1(CC(=O)N(CC(CC)NC(c2cc(OC)nn2C)=O)C)c(Cl)cnn1C Cc1ccc(C=CC(=O)N(CC(=O)NC2CC(CO)C3CC23)C2CC2)cc1 C1(C2CN(C(c3ccc(Cl)c(OC)c3)=O)C2)(NC(c2c(CC)cccc2)=O)CC1 C1(C(N2CCC(N(C(=O)C(C)(C)c3cnn(C)c3)CCC)C2)=O)CCCC(OC)C1 N1(C(C(C)NC(=O)C2CC2)=O)CCOCC1CCNC(C1(C)CCC(=O)N1)=O Cc1sc2ncnc(NCCC3CCCN(C(=O)CC4CC4(C)C)CC3)c2c1C c1(C(N2CCC(n3cc(C)nn3)C(O)C2)=O)ccc2nncn2c1.C(CO)O C1(O)(C(=O)NCC2N(C(C(F)=CC)=O)CC2)CCSCC1 c1(C(N2C(CNC(C3C(C)CC(=O)N3)=O)CCCC2)=O)ccc(N)c(F)c1F c1(C(N2CCC(C)(O)C2)=O)c(F)ccc(C#N)c1Cl C1(OCC)(CO)CN(C(=O)CNC(C2CCCCC2)=O)C1.C1(=O)C(C)N1.S(C)(=O)(=O)N Nc1nc(Cl)ccc1C(=O)NCC1CCN(C(=O)C(C2CCCCC2)O)C1 N#Cc1ccc(=NCC(=O)NCC2CC2NC(c2cc(Br)cs2)=O)[nH]c1 C1(NC(c2n(CCOCC)nnn2)(c2nnc(C3CC3)s2)C)CCOC(C(C)C)C1 Cc1nc(NC(=O)NCCCCc2ccc(F)cc2)nn1-c1cccc(F)c1 c1(NCC(CC)NC(C2(c3ccccc3C)CCC2)=O)cnc(C#N)cn1 N1(CC(C)NC(C2(N(C(C(c3cnccn3)C)=O)C)CC2)=O)CCCCC1C n1(CC(=O)NCC23N(C(CC4(CSCC)CC4)=O)CC(C2)C3)cc(C)ccc1=O C1(C(=O)NCC2CCC(C(=O)NC(c3cnn[nH]3)(C)C)C2)CC2CC(=O)C1O2 N(C(=NCCc1ccc(C)s1)NCc1cccc(Cl)c1O)CC(=C)C c1(NC(N2C(C)(CCC)CC2)=O)ccc(CC(=O)OCC)c(OC)c1 c1(C(=O)NCC2CCN2C(C2COCCO2)=O)cccnc1S C#CCC(CC(=O)NCCCN(C)OC)NC(=O)CC1CC(SC)C1 Clc1ccccc1-n1nc(CC2CC2)nc1-c1cccc(N2CCOCC2)c1 C12(C(=O)NC3(CNC(C(F)=CCC)=O)CCOC3)CCC(COC)(CC1)OC2 C1(CCCNC(c2ccc(C3CC3)cc2F)=O)CN(C(=O)C(F)C2CC2)CCO1 C1(NC(C(C)(C2CC2)OC)=O)CC(O)CN(C(=O)CCC(C)C)C1 CC1CC(NC(=O)CCSc2ccoc2)CN(C(=O)COc2ccccc2)C1 C12=CN=C(Cl)NC1=NC1CCCCC1NC2=O.C1(OC)(CF)CCC1 C1(OC(c2ccc(-c3ccc(C(=O)OC)c(C)c3)cc2)=O)CC1C1CCCCC1 CC(C)C(O)Cc1cn(CCCNC(c2cn(C)nn2)=O)nn1 c1(OC)cc(C)cc(CN2CCC3(CC2)CC3c2nn[nH]n2)c1O.C1(=O)CO1 CC(C)CCC(C(=O)NCC1COCC(C)O1)NC(c1cn[nH]c1)=O N1(C(c2c(C)oc(Cl)n2)=O)CCOCC(C(=O)NC2C=CCCC2CO)C1 N1(C(c2ccc(C(N)=O)[nH]2)=O)CCCCC(C(N2CC(N3CCNC3=O)C2)=O)C1 C1(CNC(CNC=O)=O)(CO)CC12CCN(C(c1coc(Br)c1)=O)CC2 c1(C(N2C(C)CC(NC(c3c(C)nc(CCC)o3)=O)C2)=O)cncc(F)c1Cl C(CC(C(=O)NOCC(C)O)OC)NC(CC1C(CC)C1)=O C(CC1CCC1)(CC(=O)NC(C(N)=O)C1CC1)NC(CN(CC)CC)=O.OCC CC1(C)CC(CNC(c2cccc(Cl)c2)=O)CN(C(=O)C2=CCOCC2)C1 CC1CN(C(C2(C3CCSCC3)CC2)=O)c2c(Br)cccc2S1(=O)=O C=CCC(C)(C)CC(=O)NC1(C(=O)NC(C)C(F)(F)F)CCC1 C12(C(=O)NCC3(NC(c4cc(C(N)=O)[nH]c4)=O)CCCC3)CCCC1CC2 C1(COC)(NC(=O)CCCCCSC)CCN(C(=O)C(C)(C)C#N)CC1 N1(C(C(C2CC2)OCC)=O)CCCCCCC1C(=O)NCc1n[nH]cc1C c1(OC)ccc(CO)cc1CN1CC2(CC2C(=O)Nc2ncc(CO)cc2C)C1 C12(CNC(C(COC)O)=O)CCC(CC1)N(C(C1CCC(C)=C(C)C1)=O)C2 C12CN(CCCO1)C(=O)N2.Cc1cc(Cc2nnn(C)n2)ccn1 N#Cc1nnc(N2CCC(CCCCCNC(=O)CCn3cncn3)CC2)s1 C(C(C)(C(=O)NCC(C)(F)C(C)C)NC(=O)Cn1ncnn1)SC c1(C(N2CCN(C(c3c(C)cncc3)=O)C3C2C3)=O)ncn2cc(Cl)ccc12 C1(NC(CCCC)=O)CC2(CCN(C(c3nc4cnccc4s3)=O)C2)C1 C1(NC(C(c2cnccn2)C)=O)CCC(CNC(=O)CS(=O)(=O)C(C)(C)C)CC1 C(=O)(CCCCCC#N)NCC(C(C)(C)C)NC(c1c[nH]c2ccccc12)=O N1(C(c2ccc(COC)cc2)=O)CC(C)(C)CC1CNC(C12CCC(C1)C2)=O C(C(=O)OC(C)(C)C(F)F)(C(C)C)OC(CC)=O.C1C(=O)N1 Cc1cc(=NCC2CCN2S(C)(=O)=O)[nH]c(-c2cccnc2)n1 C(CC(C(=O)N1CC(C(=O)N(C)C)C1)NC(=O)C(O)CCSC)OCC.OCC C1(C(=O)NCC(=O)OC(C)C)CN(C(C2CC(C3CC3)=NO2)=O)CC12CC2 C1(CC(=O)NCCCCC(C)NC(c2c(C)scn2)=O)CC2(CCC2)CO1 c1(C(N(CC(CNC(C(C=CC)O)=O)C)C)=O)ccnc(CC(C)C)n1 c1(CCC2NC(=O)N(Cc3noc(-c4ccoc4)n3)C2=O)ccc(Cl)cc1Br C=CCC(C)(C)C(=O)NCCn1cc(C(=O)N(C2CCC2C)C)cn1 CC1(C(=O)NCCN(CCc2ccccc2)C(c2cnns2)=O)CCC2CC2C1 Cc1cccc(-n2nc(N3CC4CC4C3)nc2C(=O)Nc2ccc(Cl)cc2)c1 C1(CC(N2CCC(C(=O)OC)C2)=O)CCN(CCc2cccnc2O)CC1 C1(C(=O)OC)CC(C(F)(F)F)CCN1S(=O)(=O)CC(C)c1ccccc1 n1(CC)cc(C(N2CCC(C)(C(=O)N(C)CC3CCCS3)C2)=O)c(C)n1 C1(NC(=O)COC2CC2)CN(C(c2cnsc2)=O)CCC1c1ccc(F)cc1 N1(C(C(CC)N(C(CSCCC)=O)C)=O)CCCCCCC1C C1(NC(CCN(C)CC)=O)CCCCN(C(=O)C(C)OC2CCOC2)C1 C(C(=O)NC1CN(C(c2ccc(C(=O)OC(C)(C)C)cc2)=O)C1)(C(C)C)NC(C)=O N1(C(c2c(CC)nn[nH]2)=O)CC(F)(F)CC1CNC(=O)CCc1ncco1 CC(C)(O)C(O)CN=c1cc[nH]cc1S(=O)(=O)NC12CCC(C(N)=O)(CC1)CC2 c1(C(C2CCCCC2)NCC(=O)NCC2N(S(CC)(=O)=O)CCC2)cccnc1O C1(CNC(c2cccc(NC(C)=O)c2)=O)CCCCCN1C(C1CC1(Cl)Cl)=O N1(C(CCNC(C2(C)C(C)(C)C2)=O)=O)CC2(CC(O)C2)C1 C1(=CC(=O)NCC(CCCC)NC(=O)C(C)c2cccs2)CCC(C)(C)CC1 C1(CNC(C2C(C)CCC2)=O)CN(C(c2ccc(NC(C)C)cc2)=O)CCCO1 Cc1cc(F)ccc1COC(=O)CNC(=O)CC(c1ccc(F)cc1)C Cn1cc(C(=O)CNC(C2CCC(n3cc(C4(O)CSC4)nn3)C2)=O)cn1 N1(C(c2nc(C)sc2)=O)CCC2(CCN(C(=O)C(C)(C)C(C)(C)O)CC2)C(C)C1 C1(NC(C2CN(C(=O)NC)C2)=O)CCC(SCCCN(C)C)CC1.C1CO1 c1(N(C)CC2(O)CCC2)nnc(C2CC2)n1CC1CCCCO1 c1(C(=O)NC(C(C(C)C)C)CNC(=O)CCCC2CC2)cc(O)cc(C#N)c1 Cc1nc(CN2CCC(C(N3CCC(C)(O)C3)=O)C2)[nH]c1C C1(C(=O)NC2C(NC(c3c(CC)nn[nH]3)=O)CCC2)CN(S(N)(=O)=O)C1 C(CCC(=O)NCCC1(C(=O)NC2CCN2c2nccs2)CCC1)N(C)CCO c1(C(=O)NC2C(C)CN(C(=O)CNC(=O)C3CC3)C2)ccc2c(n1)NCC2 C1(CNC(N2CCN(C(CC3CCCN(CC)C3)=O)CC2)=O)CCCS(=O)(=O)C1 c1(C(N2C3CCC(NC(CCC=CC)=O)(C3)C2)=O)cccc2c1OCC2 Cc1cc(=O)c(C(N2CCC2CNC(=O)C(C)(O)C2CCC2)=O)cn1C N1(C(C2C(C)(CC)C2)=O)CCC2(CC1)CCN(C(=O)C(C)C1CC1)C2 C(=O)(CC(C(C)(C)C)NC(=O)CC1CSCCO1)N1C(CC(C)C)CCC1 C1(C(N2CCC(NC(c3ccc(C4CC4)s3)=O)C2)=O)OC2CCC1CC2 Cc1nc(CN(C(=O)C(C)(C)NC(=O)CC2CCCCS2)CC2CC2)cs1 C1(CN(C)C(c2[nH]nnc2C2CC2)=O)COCCN1C(c1ncccc1Cl)=O C1(N(C(c2c(C)nsc2)=O)C)CCN(C(C2C3CCCCCCC23)=O)CC12CC2 N1(C(C(C(=O)OCC)F)=O)CCCC(C2(NC(c3cc(OC)no3)=O)CC2)C1 c1(N2CCC(CCNC(c3ccnn3CCF)=O)C2)cc(C(F)(F)F)nc(Cl)n1 c1(C(N2CCCC3NCCCC23)=O)c(F)ccc2occc12 Cc1nc(NCC2CC(CNC(=O)CC3CC4(CCC4)CO3)C2)c(C)c(C)n1 C=CCC(C(=O)NCC(O)CN(C)C(C1CC1C)=O)NC(C)=O c1(C(C(=O)NCC2(C)N(C(C3C(COC)C3)=O)CCC2)(F)F)cc(F)ccc1C C1(NC(C2CN(C)C2)=O)COC2(C1)CN(C(=O)Cc1cnco1)C2 C1(CNc2cnn(C(C)C)n2)CC2(CCC(Sc3nc4ccccc4o3)CC2)C1 C1(CN(C(=O)C(=O)NC2CCC(CN3CCOCC3)CC2)C)CC12CC(C)(C)C2 CC(C)CS(=O)(=O)CC(=O)N1CCC(OCCNC(=O)CC(O)CN(C)C)C1 c1(CC)nccn1C(C)CC(=O)NC(C)(CNC(=O)CN(CC(C)(C)C)C)CC N1(C(CC#N)=O)C2CCC1C(C(=O)NCC1(N3CCCCC3)CCCCC1)C2 c1(C(N(CCNC(C(C=C)C)=O)CC)=O)cnn2cccnc12 C(=O)(N1CC=CCO1)C1(C)CCN(C(C(COC)(F)F)=O)C1 Fc1ccc(I)c(CNC2CN(CC3CCOC3)C2)c1 C1(NC(c2cccc(CC=C)c2)=O)CCN(C(C2(COCC)CC2)=O)CC1O CCCCC(O)C(=O)N1CC2CC2(NC(c2ccc(-c3cc(O)ns3)cc2)=O)C1 C(CCNC(C1C(C(=O)OC)CC1)=O)(C(C)C)NC(=O)CNc1ccc(Cl)s1 c1(C(=O)NCCC2CCCN2C(c2ccc(Cl)s2)=O)ccnnc1Cl n1(CC(=O)NCC2CCCN2C(=O)CSCC(F)(F)F)cnc(Br)n1 c1(C(N2C(C)CCC2)=O)cnn2cc(-c3cc4ccccc4[nH]3)ccc12 CC1(C)C(=O)NCC1NC(C1(CNC(=O)C(O)C2CCCC2)CC=CC1)=O c1(NC(C(CC)CC)C)ncnc(NCCCCN2CC(C)OC(C)C2)c1C C1(COC)(CNC(c2cc3n(n2)CCC3)=O)CCN(Cc2nnn(C)n2)CC1 c1(C(=O)NC(C(CO)N(C(CC)=O)C)C)cncc(C(=O)N(C)C2CC2)c1 C(=O)(C(CCC)CC(C)C)N1CC(CC(=O)N(CCCC=C)CC)C2(C1)CC2 n1(C(c2ncoc2)(C2CC2)C2CC2)cc(CC2CC2)nn1 N#CC1(C(N2CCOCC(NC(c3c[nH]cc3C3CC3)=O)C2)=O)CC2CC2C1 C1(NC(C(C)(C)OCC)=O)CCC2(CCN(C(c3ccc(OC)cc3)=O)CC2)C1 C12(NC(=O)NCc3ccc(OC)cc3C)CCC(CC1)C(C)(C)O2 N1(C(c2c(C)n(C)nc2)=O)CCC2CCCN(C(=O)Cc3ccc(F)cn3)C2C1 OC12CCC1CN(N1CCC(c3ccon3)C1)CC2 C12(CNC(C(C)OCC)=O)CCC(CC1)N(C(=O)C(CC#N)c1ccccc1)C2 C1(C(N2CC(CC=C)(NC(=O)CC(C)(C)OC(C)=O)C2)=O)CC(=O)NC(=O)C1 CC1CCCC(C)C1n1nc(-c2ccsc2)nc1-c1cc(C#N)c[nH]1 CCCCCCCC(=O)NCC1CCC2(CCC2)C1NC(C1CS(=O)C1)=O c1(C(=O)NC2C3(CCN(C(CSCC#C)=O)C3)C2)nnc2n1CCCCC2 c1(CNC(c2c(OC(C)(C)C)cccc2)=O)nc(=N)c(C#N)c[nH]1 C1(NC(CN2CC=C(C)CC2)=O)CN(C(c2ccc(C#N)s2)=O)CC12CCC2 c1(C(N2CC(CC(=O)NC3(CO)CCOC3)(OC)C2)=O)c(F)cccc1F CC1(C)CCC=C(C(=O)NC2(CCNC(=O)Cn3cccn3)CCCC2)C1 O=C(C(O)CC(F)(F)F)NCC1C(C2CC2)CCN1C(c1cc(F)ccc1Cl)=O CCCCS(=O)(=O)NC(C(=O)NC(CN(C(=O)C(CC)N(C)C)C)CC)C(C)C C#Cc1cccc(NC(=O)NC2C(C)CCCC2C)c1 C(C1=NOC2(CCC2)C1)C(N1C(c2cn(CC(CC)O)nn2)C(C)CC1)=O C1(CCOC)CCN(C(=O)C=CCN(C)C(C2CC2C#N)=O)CC1 N1(C=O)CC2CCC1C(NC(c1nccc(C)c1)=O)C2.c1ncnc(Cl)c1F Cn1nnnc1N1CCC1C(=O)NCCN(C(C1CC(O)(C(F)(F)F)C1)=O)C1CC1 c1(N(CC(=O)NCCNC(c2c(C)onc2O)=O)C)ccc(Cl)cc1C#N CCCC(C(=O)NCCOCCNC(C1CC12CCOC2)=O)OC C1(CNC(c2c(C)nns2)=O)COCCN(C(=O)CCC2CCN(C)CC2)C1 C1(NC(C2CC23CCC3)=O)C2CC3C1C3C2C(=O)NC1CC2CCC(C1)S2 CC(C(F)C(=O)NCC1(O)CN(C(c2ccc([N+](=O)[O-])c(O)c2)=O)C1)C(F)(F)F c1(OC)cccc2sc(-c3nc(-c4ccsc4)nn3CCOC)cc12 C1(C(N(C2CC2)NC(C#C)C)=O)CCC(F)C1.C12(CCC1)N(C)C2=O.CC N1(C(CCSCC(C)C)=O)CCN(C(C2CCC2)=O)CC1C1CCC1 C(=O)(C1c2ccccc2C2CC1C2)N(CCC)CCNC(=O)C(C)SC c1(C(=O)NCC(CC(=O)NCC2CC3CCC(C2)C3)OC)cn2ccccc2n1 C1(C(=O)NC(C2C(C(=O)NC(c3nc(C)[nH]n3)(C)C)C2)C)C2CCC(C2)C1C C=CC1CCCCN1C(=O)C(C(C)OC)NC(=O)CCC(N)=O C1(CCC)CN(C(=O)Cc2cnc[nH]2)CC1NC(=O)CCCc1ccncc1 C12CCCN(C1)CC(=O)NC2.n1(CC(N2CC(CC)C2)=O)nnc(=O)[nH]1 c1(OC)cc(Br)ccc1C(N1CC=CC(NC(=O)CN2CCCC2=O)C1)=O c1(CC(C)C)cc(C(=O)N(C(C)CNC(=O)Cn2nccn2)C)cc(O)n1 C1(C(=O)NC(C(CC)OC)C2CC2)C=CCN(C(C2(CC)CCOC2)=O)C1 C1(C)(CNC(c2nc(C(C)C)oc2)=O)CCCN1C(c1n[nH]c(C(C)(C)C)n1)=O N1(C(C(C2CC2)NC(CN(CCOC)C)=O)=O)CCCOCC1C Cc1sncc1C(=O)NCC(C1CCCCC1)NC(=O)CCn1cc(Cl)cn1 Cn1ncc(Br)c1C(N1CCC1CNC(C1(C(F)(F)F)CC=CC1)=O)=O C(=O)(CC(C)(C)C(F)F)N1C(CN(C(COCC#C)=O)CC)CCCC1 C=CCN(OC)C(=O)CCC1CC(NC(C2CC2Cl)=O)C1 N1(C(c2cc(C)[nH]n2)=O)CC2CC(NC(=O)CC3CC4(CC4)CO3)C1C2 C(=O)(CC(C(F)(F)F)OC)NC1(C)CCCN(C(c2cc(OCC)n[nH]2)=O)C1 c1(C2(C(=O)NC3C(NC(COCCSC)=O)CCC3)CCC2)ccc(F)c(Cl)c1 C1(CCC)CN(C(=O)Cc2ccco2)CCN1C(=O)CC1COCCN1C c1(CC(=O)OCC)cc(F)ccc1S(=O)(=O)N1CCN(CC(=O)OC(C)(C)C)CC1 C1(NC(C2CCOC2)=O)COCCN(C(=O)C(F)=CCCCC=CC=C)C1 C1(SC(F)F)CCCC(NC(=NCc2ncccn2)NCCc2nccs2)C1 c1(OC)ccc(C)c(OC)c1C(N1CC(NC(c2ncncc2Cl)=O)C1)=O N1(C(C(C)OC)=O)CCC2(CCC(NC(c3cc(C)nc(O)c3)=O)CC2)CC1 c1(C(N2CCC(CNC(C3(C)C(C)C3)=O)C2)=O)c(N)cc(F)cc1Cl c1(-c2n(C(c3ccccc3)C)nc(-c3ccsc3)n2)ccc2c(c1)nnn2CCOC N1(Cc2cccc(OC)c2C)CCC(NC(=O)Cc2ccccc2F)C(C)(C)C1 c1(SC)cc(C(=O)NCCC(C)N(C)C(c2sc(CO)nc2C)=O)c(C)o1 N1(C(C(C)OCC)=O)CCC(CC(=O)N(C2CCC2)CCO)CC1 Cc1cnc(NC2(C3CC3)CCOCC2)c(S(=O)(=O)NC(C(C)C)C2CCC2)c1 Cc1cc(C(N2CCC(C3CCCN3C(c3coc(Br)c3)=O)C2)=O)c(C)n1C CCCCN=C(NCCF)NCC1CCS(=O)(=O)N1C C=CC(CCC)CC(=O)NCC(CCC)C(=O)NC1CCCCC1(C)O CC1CCc2nc(C(=O)NCC(F)(F)F)cc(N3CCC(O)(C(C)(C)C)C3)c2C1 N1(C(C(C=C)O)=O)CCC(CCOC)(NC(=O)COCC2CC(F)(F)C2)CC1 C(=O)(C(C)CC(F)(F)F)NCC1(F)CCN(C(C=CSC)=O)C1 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCCC(CCNC(CCCOC)=O)C C(=O)(C1=NOC(c2ccccc2)C1)NCC1(CO)CCCC1.C12(CC1)C(=O)N(C)C2 CC(O)C(C(=O)N1CCC(O)(CCNC(=O)CCCc2ccccc2)C1)N(C)C c1(C(N2CC(C(C)NC(C(CC)n3ccnc3)=O)C2)=O)cn2ccnc2cn1 C(C(C)(C)C(=O)N1CCC(CC(=O)Nc2ccc(C(=O)C(F)(F)F)cc2)C1)OC CCC(C#N)(CC)C(=O)N1CC=CC(NC(=O)C=CSc2nc[nH]n2)C1 c1(C(N(CCN(C(c2c(C)nccn2)=O)C)C)=O)ccc2ccnc(O)c2n1 c1(C(=O)NC(C2CC=CCC2)C(N2C(COC)C=CC2)=O)cn(C)c(=O)cn1 c1(C(C)C)c(C(N2CC3CC3(C(=O)NCc3ccc(F)nc3)C2)=O)cnn1C C1(C(N(CCC)C)=O)(C(C)C)CCN(C(=O)Cn2ccc(C)c2)C1 c1(C(=O)NCC2CN(C(C(CCSC)NC(N)=O)=O)CC2O)cnc2sccn12 C1(C(N2CC(COC)(CNC(c3cc(Cl)cnn3)=O)C2)=O)OCCOC12CCC2 C1(CNC(C2CCC(O)C2)=O)CC2CCC1N(C(c1cncc(Br)c1)=O)C2 c1(CC)cc(C(=O)NCC(CO)NC(=O)C(C)C(=O)N2CCOCC2)c(C)o1 CC1CN(CCN2CCCC2)CCN1N1CCC(c2ccc(F)cn2)CC1 c1(C2(C)C(=O)N2)cccc(Cl)c1.N1(CC(C)NC(=O)C(=O)N(C)C)CCCC1 Cc1[nH]c(C(C)(C)C)cc1NC(C1CCC(COC(F)(F)F)O1)=O N1(C(c2cc(CC)no2)=O)CCC2CCC(C1)N2C(=O)CC(O)CN(C)C Cc1cc(C(N2CCC(F)(C(N3CCOC(C#N)C3)=O)CC2)=O)cc(C)n1 C(=O)(C(C(C)O)NC(N)=O)NC(C)C(CO)NC(c1ncncc1F)=O C(=O)(C1=C(C)N(CC)C(=O)NC1c1ccc2c[nH]nc2c1)NCC(=C)C c1(C(N2CCN(C(C(=O)NCCC)C)CC2)=O)cc(F)cc(F)c1 CCC(C#N)C(=O)N(O)Cc1cn(Cc2nn(C(C)C)cc2C)nn1 C1(NC2CC(OCC)C2)CCN(C(c2cnnn2CC)=O)CC1C c1(C(C)C)ccc(NC(C2CN(Cc3ccc(CCBr)cc3)CC2O)=O)cc1 C(=O)(C1CCc2c(Cl)cccc21)NCC(C)N(C(Cc1c(C)noc1)=O)C C1(CNC(Cc2cn(C)nn2)=O)(CO)CCN(C(=O)CCCc2cc[nH]n2)CC1 C1(C(N2CCC(NC(=O)CCc3ccoc3)C2)=O)CCCc2ccccc2C1 C1(C(C(=O)NCCC(=C)CNC(=O)Cc2cccc(C)c2)C)CCN(OC)CC1 c1(NC)ccc(C(N2CCC(NC(=O)Cc3scnc3C)C(F)C2)=O)c(Cl)c1 C=CCC(C(=O)N(C1CCCN(C(=O)COCC(=C)C)C1)C)N(C)C N1(C(C=CC(C)(C)NC(C(C)CCN(C)C)=O)=O)C2CCC1CC(F)C2 CC1(CNC(=O)CC2CCCCC2NC(c2ncccc2F)=O)CCCCCC1 c1(NC(C(CC)C)(C)c2nnnn2CC)ccc(-c2ncn(C)n2)c(Cl)c1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC1(C)C(=O)NC(c1cccc(C)c1)CO c1(C(N=c2ccn(C)[nH]2)=O)n[nH]c2ccc(-c3cnn(CC#N)c3)cc12 Cc1ccc(NC(=O)CCCCCNC(C2CC(C)(O)C2)=O)cc1O N1(C(c2occ(C)c2)=O)CC(O)(C2CCN(C(C3CC4CCC4C3)=O)CC2)C1 Cc1cc(C(N2CC3CC(NC(=O)C(C)C(C)O)C3C2)=O)cc(N)c1 c1(CC(=O)NC2CCN(C(C(COCC)C)=O)C23CC3)c(C)nc(O)nc1O C1(F)(C(=O)NCCN(C)CCO)CCCN(C(=O)CCS(N)(=O)=O)C1 CC12CC(C(=O)N(C(=O)Cc3cccnc3)CCCO)(C1)C2.C1CC1 c1(CCN)ccc(-c2nc(-c3ccc(Br)cc3)n[nH]2)cc1 C(CCF)(C(=O)NCC1(O)CC2CC1C2)NC(=O)Cn1cnnn1 C(=O)(CCCC(=O)N1CC(NC(c2c(C)noc2C(C)C)=O)CC1C)NCC Cc1ccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC(C(C)(C)O)C2CC2)c(F)c1 CC1(C)OC2(C(=O)NC3CN(C(=O)CCc4ccc(Cl)cc4F)C3)CC1C2 C1(NC(c2cncnc2)=O)CCN(C(=O)C(O)CC2CCCCC2)C1C1CC1 c1(C(CNC2CCOC2)NC(=O)Nc2c(CC)onc2C)c(C)cccc1Br C(C1=CCN(C(=O)C(S(C)(=O)=O)C2CC2)CC1)NC(CCCc1c(C)[nH]nc1O)=O CC1CCc2cc(C#N)c(N3CC(CCCCNC(C4CC4(C)CF)=O)C3)nc2C1 c1(CNC(c2c3c([nH]n2)CN(C(C)=O)CC3)=O)ccc2c(c1)C(=O)N(C)C2 N1(C(C(C)(C2CCC2)NC(c2c(CCC)nco2)=O)=O)CCOC(C)(C)C1C C1(CC(=O)NC2(CNC(c3c(OC)nsc3)=O)CCC2)CCC(=O)NC1 CCC(C(=O)NC1CCC(CNC(c2coc(C)n2)=O)C1)N(C)C c1(C(N(C2CCN(C(=O)CCF)CC2)CCOC)=O)ccc2c(c1)CCC2 N1(CC(=O)N(CCCNC(c2ccc(NC3CC3)nc2)=O)C)C(=O)CNC1=O N1(C(Cc2cc(C)no2)=O)CCCC(C(=O)NCC(c2cccnc2)O)C1C C1(NC(c2coc(-c3cccnc3)n2)=O)Cc2cscc2C1 c1(NC(C)=O)ccccc1Br.c12nc(cs1)C(=O)NC2CC c1(C(=O)NCC2C(NC(CC(C)CN(C)C)=O)C2)ccc2cc(F)ccc2n1 C(=O)(C(O)CC(C)(C)C)NCCC(CNC(c1c(C)n[nH]c1C)=O)O c1(C(=O)NCCn2cc(C(=O)NCCO)nn2)cc(F)cc2c1NCCC2 N1(C(C(C2CCCC2)OC)=O)CCC(C2CC2)(NC(c2ccns2)=O)C1 c1(CC)ncccc1C(=O)NCC1CCN1C(=O)Cc1ccccc1F C1(NC(c2c(CC)occ2)=O)CCN(C(=O)CSCCOC(C)=O)C(C)C1 N1(C(C2N(C)CCCC2)=O)CCC(C(=O)NCC2(CCCO)CC2)C(C)(C)C1 c1(C(=O)NC2CCC(NC(c3ccc(C)c(CO)c3)=O)C2)cc2c(cn1)OCO2 Cc1ccc(C(N2CC(NC(c3ccc(I)cc3)=O)CC(C)C2)=O)c(F)c1F n1(CC)nc(C(N2CCC(NC(c3ccsc3OC)=O)C2CC)=O)cc1C1CC1 N1(c2n(CCCOC)c(-c3cc4c(s3)CCC4)nn2)Cc2ccc(O)cc2C1 C1(NC(C(CC)C)=O)C=CCN(C(c2cc(-c3ccc(Cl)cc3)no2)=O)C1 C=CCC(C(=O)NCC1CC(C)(C)CN1C(c1ccn(C)n1)=O)C(C)C C1(C(=O)NCc2cc(C)ncc2)CN(C(c2cc(Cl)cs2)=O)C(C)(C)C1 C1(NC(C=CC(=O)N(C)C)=O)CN(C(c2cc(N)c(F)cn2)=O)C2(CCOCC2)C1 N1(CCCNC(C=C(C)C)=O)CCN(C(=O)C=C2CCN(C)C2)CC1 Cc1cc2c[nH]nc2cc1C(N1CCCN(C(=O)CC2CC=CCC2)CC1)=O CC1=NOC(C)(CNC(=O)C(=O)NCCC2(C)CCCO2)C1 C(=O)(CN=c1[nH]c(C)cs1)N1CC(F)(CNC(Cc2nc(CC)sc2)=O)C1 C1(C)(CC)CCCN(C(C2CC(CNC(c3cncc(C)n3)=O)C2)=O)C1 C1(C(=O)NCC(C(=O)OCC)(C)C)CC2(C1)CN(C(C1(COC)CC1)=O)C2 c1(CNc2ccc(C(N(C(CC)C)CCO)=O)cn2)cnc2cc(C)nn2c1 C(C(CC(F)(F)F)NC(C1CCCOC1c1ncc[nH]1)=O)NC(C12CC(C1)C2)=O Cc1ccc2ncc(C(N3CC(NC(C4(C)CC(C#N)C4)=O)CC3C)=O)n2c1 c1(C(=O)NC(CN(C(C2C(CC)OCC2)=O)C)(C)C)cn2ccnc2cn1 c1(C(C(=O)NC(CC)(C)C)N(C2CCCCC2(C)C)C)n[nH]c2c(Cl)cccc12 Cc1cn2cc(C(=O)N(C)CC3CCCN3C(C3(C)CCCC3C)=O)sc2n1 C1(NC(Cn2cc(C(=O)OCC)nn2)=O)CCOCC1NC(c1cnoc1C)=O c1(C(N2CC(O)(C(C(=O)NCCC=CC)F)C2)=O)ccn(CC)c1C N1(C(C=CC=CCCCCC)=O)CCN(C(c2cc(C)sc2N)=O)CC1 N12CCOCC(C1)C(=O)Nc1ccc(o1)CCNC(=O)C2.O=CN.C(=O)(C1CC1)N c1(C(=O)NCC2(F)CC(NC(CCC#C)=O)C2)ccccc1CC=C N1(C(C(=Cc2ccncc2)C)=O)CCC2CCC(NC(c3ccncc3)=O)C12 CN1CCN(C(C2CC3COCC3C2)=O)C(CNC(c2n[nH]cc2[N+](=O)[O-])=O)C1 n1(Cc2cccc(C3(C)COC3)c2)cc(C#CC(C)(C)NC(=O)CN)nn1 c1(C(=O)NCCC2N(C(COCCCC)=O)CCCC2)cc(F)c2c(c1)CCC2 CCCC(C)(O)CC(=O)N1CCCC1(C)CNC(c1n[nH]c(C)c1Br)=O c1(C(=O)NCC(C)(C)NC(C=CC)=O)ccc(=O)n(CCO)c1 C1(C(=O)NC(CNC(C(CC)N(C)C)=O)C2CC2)(CF)CCOCC1 C(C(F)(F)C(F)F)NC(C1(n2cc(CC(O)CNC3CC3)nn2)CCOCC1)=O CCCCC(CC)CC(=O)NCC1CCCCC1NC(=O)COC(C)(C)CC CCCCCC(O)C(=O)N1CC(NC(c2nnc(C)cc2O)=O)CC(C)(C)C1 C1(N(C(=O)COC2CCCOC2)C)CCCN(C(=O)CCc2ccco2)C1 Cc1oc(C(C)(C)C)cc1C(=O)NCC1CCCN1C(N)=O N1(C(c2ncccc2Cl)=O)CCCC(C2CC2NC(C2CC(CC3CC3)C2)=O)C1 C1(CNC(C)=O)CCC(NC(C2CCOC(C)C2)=O)CC1 C1(C(=O)NCCCC2(NC(C(CC)F)=O)CC2)CCC2(CCC2)O1 Cn1cc(C(N2CC3CC3C2C(N2CCCC(C(N)=O)C2)=O)=O)ncc1=O c12ccccc1C(=O)N2.N1(C(=O)NCCC)CCN(CCC)CC1 c1(C(N(CCCNC(c2cc(C)sc2C)=O)CC)=O)[nH]c2ccc(F)cc2c1C C(=O)(C(O)CC(C)(C)C)N1C(CNC(C(c2ccc(F)c(F)c2)C)=O)CC1 C(c1ccc(F)c2ccccc12)=CCN(C(C#C)Cc1ccc(F)cc1)C1CC1 c1(N(C(CN(C)CCc2nc(-c3cccs3)n[nH]2)=O)C2CC2)ccc(F)cc1 C(=O)(CC(C(=O)N(C(C)(C)C)C(C)C)N1CCNCC1)OC.C1(=O)C(C(C)C)N1 CC1(NC(=O)CC2(C)CCCO2)CN(C(C2CCC(=O)O2)=O)C1 N(C1COc2cc(Br)cc(F)c21)C(N1CCCC(F)(CO)C1)=O c1(C(=O)Nc2nc(Cl)ccc2I)ccc2c(C(=O)N=c3cco[nH]3)n[nH]c2c1 N1(C(=O)C2=COCC2)CCCC2(CCN(C(=O)C3COc4ccc(F)cc43)C2)C1 C1(NC(C2(C)CC=CCC2)=O)CC2(CCCCN2C(=O)CCC2CC2(F)F)C1 C(C(C(=O)N(CC(C)O)CCOC)C(C)C)NC(c1n(CC)nc(C)c1)=O C=CC(CCC)CC(=O)NC1CCCCC1NC(c1cnn2ncccc12)=O C=CCC(CNC(C1C=C(C)CS1)=O)C(=O)N1CC(n2cnnc2)C1 CC1=C(C(=O)NC(c2c(C)n[nH]c2C)(C)C)CCO1.C12CCN(CC1)C2=O c1(SC)cc(C(=O)N(CCCNC(C2C=CCCC2)=O)CCO)oc1C n1(CC(=O)NCCCN2CCN(C(C3N(CC)CC3)=O)CC2)cc(F)ccc1=O c1(C(=O)NCCOCCNC(c2n[nH]c(C)c2O)=O)cc2cscc2s1 c1(C(=O)NCC(C)NC(=O)CCC2CCCN2C)coc2c1C(O)CCC2 c1(COC(C(CCC)OC)=O)ccc(Cl)cc1Cl.c1(C2C(=O)N2)ccccc1 c1(C(CO)NC(=O)CNCCC2CC2(Cl)Cl)ccc2c(c1)CCC2 C1(CC)CN(C(c2ccc(F)c(NN(C)C)c2)=O)CCN1CC(F)F C1(N(C(c2cccc(OC)c2F)=O)C)CC2CCC(C1)N2C(=O)CCC(F)F Cc1nn(CC(N2CC(CNC(C3CC3CF)=O)C(O)C2)=O)cc1Br c1(C(=O)NCC2CC(NC(C3(COC)CC3(F)F)=O)C2)ccc(C)c(F)c1 C1(C(=O)NCC(CNC(=O)CCc2ncccn2)OC)(CSC)CCOCC1 c1(SC)cc(C(=O)NC(C)CC2CCCO2)ncn1.C1=CCNC1=O C1(C(=O)NCCCCCN(C(C2(C(C)C)CCCO2)=O)C)CC(=O)N(O)C1 C1(C(=O)NCCCOCC#C)CC2(CCC2)CN1C(c1cnc(O)cc1O)=O N1(C(Cc2ccc(C(N)=O)cc2)=O)CC2CCN(C(C3CCCOC3)=O)C2C1 C1(C(=O)NCC2N(C(C(C)C3CCC3)=O)CC2)CC2CC1C1C2C1(F)F c1(OC)ccc(CCNC(N2CCC(C#N)C2)=O)cc1I c1(NC(COCCNC(c2ccc(C(C)=O)[nH]2)=O)=O)ccc(Cl)cc1O C(=O)(CCC1=CCCCC1)N(C1CCN(C(C(CCC)OC)=O)C1)CC1CC1 Cc1ccc(C#N)c(N2CCC(CNc3scnc3C3CCCCO3)C2)c1 N1(C(CC(C)n2cccn2)=O)CCC(C2CC2)C1CNC(C1(O)CCSCC1)=O N1(C(C)=O)CCN(C(C2CC2(C)C)=O)CC2(C)CCCC12 c1(C(=O)NCC(CSCC)(C)C)ccc(C2CC2)cc1Cl c1(CC(=O)NC2CCN(C(C(CC=CC)CC)=O)C2)nn(C)cc1[N+](=O)[O-] C(=O)(C#CC(C)(C)O)N1C(C(N(CC(CC)(O)CC)C2CC2)=O)CC(O)C1 c1(CC)c[nH]cc1C(=O)NCC1CC(NC(=O)Cc2csc(C3CCCC3)n2)C1 Cc1ccc(C(N2CCC(CCNC(=O)C(O)C(C)C)CC2)=O)c(Br)c1F CCC(CCC(=O)NC(c1cscn1)C)NC(c1ccc(C(C)C)o1)=O C1(C(N2C(C3CCN(C(c4ocnc4C4CC4)=O)C3)CCC2)=O)CCS(=O)(=O)CC1 CCCCC(CNC(=O)CCCOCCC)NC(c1n[nH]cc1Cl)=O NS(=O)(=O)CC(=O)NC12CC(CNC(c3cncc(OC(F)F)c3)=O)(C1)C2 c1(C(=O)NCC2CCN(Cc3onc(CCC)n3)C2)cnn2ccn(C)c12 c1(C(=O)NC(C)CNC(C2CN(C3CCCCC3)C2)=O)cnc(C(F)F)cn1 N1(C(CSCCN(C)C)=O)CCC(CNC(=O)CC23CCC(C)(C2)OC3)C1(C)C C(=O)(CC(F)(F)C(F)F)NCC1C(C)(C)C1C(=O)NCC12CCN(CC1)CC2 c1(NC(CCCCCCC2CCCCC2)=O)cccc(-c2cn(C3CC3)nn2)c1 n1(CCC(=O)NCCCSCCCO)c(=O)oc2ccccc12 C1(N(C)C(c2cnc(S)n2C)=O)CCCN(C(=O)CC=C(Cl)Cl)CC1 c1(NC(=O)NCc2nc(C(F)F)no2)ccc(F)c(Cc2cccnc2)c1 n1(COC)ncnc1C(=O)NCC1(NC(c2ncoc2-c2cc(C)no2)=O)CC1 c1(C(=O)NC(CC)CNC(=O)Cc2cn[nH]c2)oc(P(C)(C)=O)cc1C c1(C(=O)NC2CC(NC(CC3(C)CC3(Cl)Cl)=O)C2)cnn2c1OCC(O)C2 c1(CN(C(=O)CN(C)C(C2CC2F)=O)CC#C)cccc(O)n1 CS(=O)(=O)c1ccc(CCNC(C2CCN(Cc3ccccc3)C(=O)C2)=O)cc1 N1(C(CCCC)=O)CCC2(CCCC2NC(c2cc(O)ncn2)=O)CC1 N1(C(=O)C=CCN2CCOCC2)CCN(C(C2CCCC3CC23)=O)CC1 c1(C(N2CC(n3cc(CNC(C4CCC(C)O4)=O)nn3)C2)=O)ccnc(F)c1F c1(C(N2CC(CNC(C3CC4(CCC4)C3)=O)OCC2)=O)ccc2ncsc2c1 Cc1cccc2cc(NC(C3CC4CC3CN4C(c3n[nH]c(=N)[nH]3)=O)=O)sc12 C1(CC(N2CCC2c2cn(-c3cccc(Cl)c3)nn2)=O)CCS(=O)(=O)C1 C(=O)(C(C1(C)CC1)NC(=O)CCc1cnn[nH]1)NCCOC(C)C N1(C(C2(CC)CC2)=O)CCC2CCCN(C(c3ccc4oc(C)cc4c3)=O)C2C1 C(CCO)(C(=O)N1CCCC1C1(NC(=O)Cc2cnccc2Cl)CC1)N(C)C Cc1ccc2c(OCCCOc3cccc(Cl)c3)ccnc2c1 c1(CN(C(CC2(OC)CCC2)=O)C)ccccc1CNC(=O)Cc1n[nH]c(C)n1 c1(CC)cccc(C(=O)NCC2C3CN(C(=O)C(C)(C)OC(C)C)CC23)n1 N1(C(C(c2c(C)cccc2)C)=O)CC(NC(c2cc[nH]c2)=O)C2CC2C1 c1(CN=C(NCCC=C)NCC2CC2OCC)ccc2c(c1)n(C)c(=O)n2C c1(OC)ccc(S(=O)(=O)N2CCC(CNC(c3ccc(Br)nc3C)=O)C2)cc1OC C#CCC(CC#C)C(=O)NCC(CC=C)NC(=O)COc1ccc(F)cc1F C1(O)(CNC(c2c(C)noc2N)=O)CCCN(C(C2CC23CC(C)(C)C3)=O)CC1 CC(CN=c1ccc2ncc[nH]c-2n1)N(C)C(C1CCc2ncnn2C1)=O C1(C)(CCNC(C2(OC)CC(C)C2)=O)CCN(C(=O)C(C)(C)C2CCCCO2)C1 N1(C(CC(CC=C)(C)C)=O)CCCC2CN(C(=O)C=CC(=O)N(C)C)CCCC12 C#CCC(O)C(=O)N1CCCCC1CCNC(=O)C(N1CCOCC1)C C1(NC(C2CN(S(N)(=O)=O)C2)=O)COC2(C1)CN(C(C1CC1C(F)F)=O)C2 C#CCCC(C(=O)Nc1cccc(C)c1)NC(C1C(C)(C)C1(F)F)=O N1(C(CCOC)=O)CCC(CCNC(c2ccsc2Br)=O)CC1C Cc1ncccc1C(N1CC(NC(=O)C(c2cccnc2)C)C1)=O C(=O)(CC(CN(C)C)C(F)F)NC(c1ccccc1)CNC(C(COC)OC)=O C1(C(=O)NC(CCC)C2CCC2)CCCN(C(=O)CNC(=O)OC)CC1 C(CCC(=O)NC(C)CCNC(C1(C(C)(C)C)CCCC1)=O)OC(C)C C1(CNC(CCOC(C)=O)=O)CN(C(=O)COc2ccc(C#N)cc2)CCC1C N1(C(c2c(C)cn(C)n2)=O)CCN(C(C2(C)CCCCC(C)C2)=O)C2(CC2)C1 C1(NC(c2cn(-c3cnn(C)c3)cn2)=O)CCN(C(=O)Cc2ccc(Cl)s2)C1 CN(Cc1ccc(OC(C)(C)C)cc1)N1CC(Cc2cnccn2)C1 CN1CCn2cc(C(=O)NC3(CNC(=O)Cc4cnn(C)c4)CCC3)nc2C1=O c1(CNC(C2CCN(c3nnc(CO)s3)CC2F)=O)nnc2n1CCCC2 N1(C(c2c(C(C)=O)cnn2C)=O)CCC(NC(c2ccsn2)=O)CC(C)(C)C1 CC(C)C(C)(C)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1cnn(C)c1 c1(C(=O)NC2CCCCN(C(c3cc(C)c(C)o3)=O)C2)ccc2ocnc2n1 C1(C(N2C(CNC(CC3(C)CC3)=O)CC3(CC3)C2)=O)CC2CCCC(C1)C2 N1(C(C(C)OCCN(C)C)=O)CCOC(CCNC(C2CCC3CC23)=O)C1 c1(C(=O)NC(CNC(CCCC(CC)(C)C)=O)(C)CO)cc2ccc(Cl)cc2s1 C(=O)(CCCC(F)(F)CO)N1CC(NC(CC2(NC(C)=O)CC2)=O)C(C(F)F)C1 C(=O)(C(O)C(F)(F)F)N(C(C)C(=O)NC1CC=CCC1)C1CC1 CC(C)CC(CN=c1[nH]c2ccc(Cl)cc2s1)NC(=O)CCN1CCCCCC1 C(C(C)(C)C(=O)N(C12CCC(CC1)O2)CC)NC(c1nc(OCC)sn1)=O.COC Cc1c(C(N2CCC(NC(c3cccc(F)c3)=O)C(F)C2)=O)ccc2c1CCC2 c1(C(=O)NC2CC3(CN(C(c4cc(OC)no4)=O)C3)C2)cc2c(cn1)OCCO2 C(C(CC(F)(F)F)NC(=O)OC(C)(C)C)NC(C1(NC(C(C)C)=O)CCCO1)=O Cc1cccc(C(=O)NCCC(C)NC(=O)C(C)CC2CC2)c1C#N C1(CNC(CC=CCCCCC)=O)CCCN(C2CCN(CC(C)C)C2=O)C1 C#Cc1ccc(F)c(C(=O)N(C2CN(C(C3CC(N(C)C)C3)=O)CC2O)C)c1 C=CC(CC)CC(=O)NC1(CCOC)CCN(C(C2CCN(C)C2C)=O)CC1 C12CCCCC1NC(=O)CONC2=O.CC1(N(C2CC2)C2CC2)CC1(F)F N1(C(C(C#C)(C)C)=O)CCCC2(CCC(NC(c3ccc(Cl)cc3)=O)C2)C1 c1(NC2C(c3n(CC)ccn3)OCC2)cc(CNC(=O)OC(C)(C)C)ccc1O CCCCC(CC)C(=O)NC(CNC(=O)C=CCOC)C1CCC1 c1(C(=O)NCC(C)(C2CC2)NC(C2CC3CCC2CC3)=O)coc2ccccc12 CCCCC(CC(=O)N1CCC(O)(C(N)=O)CC1)NC(C1COCC(C)O1)=O c1(SC)ccc(C=CC(N2CC(NC(=O)CC(C)(C)C)CC(F)C2)=O)cc1 C1(OC)CCN(C(C2CN(C(=O)Cc3cc(C)on3)CC2(F)F)=O)CC1(C)C CC1CN(C)CC1NC(c1c(CNC(=O)CCc2cnoc2)cnn1C)=O c1(C(N2CCC(C)(CNC(c3n(CC)ncn3)=O)C2)=O)cc(C(C)C)nc(O)c1 CC(C)(CC(=O)NCC1(C2CC2)CCN(C(C2CCCC(O)C2)=O)C1)C(F)(F)F C1(NC(CC2N(C)CC=CC2)=O)CC=C(C(=O)NCCn2cccn2)C1 C1(C(N2CC(O)(C(C(=O)NC(CC3CC3)C3CC3)F)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(C(N)=O)cc1C(N1CCOCC1Cc1cnoc1)=O CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cc(C)n(C4CC4)c3C)=O)C2)CC1 C=C(C)CCCC(=O)NCC1CC1NC(=O)Cc1sc(-c2ccn(C)n2)nc1C N1(C(C2C(C)C2)=O)CCC(C2CCN(C(c3ccc([N+](=O)[O-])n3C)=O)C2)CC1 CCC(C(=O)N1CCC(NC(=O)Cc2cncnc2)C(O)C1)C(C)(F)F C(CC(C(=O)N1CCC1CC(C)C)NC(=O)C1=NOCC1)NC(C)=O c1(CC)ccc2nc(CC(=O)NC(Cc3ccncc3)C(=O)O)cn2c1 c1(C(=O)NC2CCCC(N(C(CSCC#C)=O)C)C2)c(C)cc(OC)cc1F C=CC(C)(CCOC)C(=O)NCC(C)NC(=O)Cc1c(C)cc(N(C)C)cc1C C1(CC(=O)NCC2N(C(Cc3scc(C)c3)=O)CCCC2)CCn2cncc2C1 CN1C(=O)CCc2c(C(=O)NNC(=O)C(C)(F)c3ccccc3)cccc21 N1(C(C(CCC)C)=O)CCN(C(c2ccc(CF)cc2)=O)C2CCCC12 c1(NCc2ncc(C)c(OCC)c2C)ncc2c(n1)CCC(C(F)(F)F)C2 C(=O)(C1COc2ccccc21)NCCCC(C)NC(C(CC)OC)=O C#CCC(C(=O)NCCC(O)CCO)NC(c1cnncc1O)=O N1(C(c2cc(C(C)(C)C)sc2)=O)CC(F)CC1C(N1CCC(CO)C1)=O C1(NC(C2(OC)CCCSC2)=O)CCN(C(c2c(C)ccn2C)=O)CC1CO N1(C(C=CC)=O)CCCC(NC(C2CC(=O)NC2(C)C)=O)C1C c1(-n2c(-c3cnc(Br)o3)nc(C(C)OC)n2)ccc(Cl)cc1OC(F)F C1(CNC(=O)N(c2scc(-c3c[nH]c(=N)s3)n2)C2CC2)CC2(CCNCC2)C(=O)O1 CCC1=NOC(CC(=O)NCC(=O)NC2CC23CC(NC(=O)CC(Cl)Cl)C3)C1 Cc1coc(C(=O)NCC(C)(C)CNC(=O)C(C)Cc2ccccc2)c1 N1(C(C(C)(c2ccccc2)N(C)C)=O)CCC(NC(C2CC=CC2)=O)C(O)C1 c1(CN2CC3C(C(=O)NCC(C)C)(C3)C2)cccc(F)c1C#N c1(C(N2C(C)CN(C(=O)CC3CCC3)CCC2)=O)cc2c(nc1O)CCCC2 c1(OC)cc(Br)c(C(C)NCc2nccs2)cc1OC C(=O)(C(N)C[Si](C)(C)C)NC(C1CCN(C(C)C)C1)=O c1(C(N2CCCC(c3cn(CCS(CC)(=O)=O)nn3)C2)=O)csc2nccn12 C(=O)(C1=CS(=O)(=O)CCC1)N1CC(C)N(C(c2ncn(C)n2)=O)CC1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1)NCCN(C(=O)CN(C1CC1)CC)CC C(c1ccc(F)cc1)=CC(N1C(C2N(C(c3ncn(C)c3)=O)CCC2)CCC1)=O N1(Cc2cn(CCC)nc2)CCC(F)(F)C(NC(c2cc(C)cc(O)c2)=O)C1 c1(C(=O)N(CCC2(NC(CSC(C)(C)C)=O)CC2)C2CC2)c(F)cc(Cl)cc1F Cc1cc2cc(C(=O)NC3CCCN(C(=O)CC4CC5(CC5)C4)C3)ccc2cn1 Cc1nc(C2CC2)sc1C(=O)NCC1CC2CC2N1C(=O)Cc1cccn1C Cc1ccc(OCC(=O)NCC2CCCN2C(=O)CN(C)C(C)C)c(Br)c1 c1(COC)ccoc1C(=O)N(CCCCCNC(C1CC(COC)C1)=O)C N1(C(C(C)OCCC=C)=O)CCCCC1C(=O)NC1(C)CSC1 c1(CNC(C(C)OC(C(CSC)C)=O)=O)cccc(Br)n1 C(COC(C)C)(C(=O)NCC(C)NC(C12CC(CO1)C2)=O)NC(C)=O c1(C(=O)NCC2(NC(COCC(=C)C)=O)CCOCC2)cc(Cl)c2n[nH]cc2c1 C1(CCNC(CCC=C)=O)CCN(C(=O)CCC2CCC(=O)N2)CC1 c1(OCC(N2CC(C(=O)O)CC(OCC)C2)=O)ccc2cc[nH]c2c1F c1(CC(=O)NC(CNC(COCCC=C)=O)CC=C)ccc(O)nc1 c1(C(=O)NCC2(C)C(C)CN(C(COC(CC)C)=O)C2)cc2cc(Cl)ccc2[nH]1 c1(C(=O)NCC(C)CNC(=O)C(F)CC2CC2)nc[nH]c2nccc1-2 CS(=O)(=NCC(=O)NC(Cc1cccc(Br)c1)C(F)(F)F)C1CCOC1 N1(C(c2c(CC)nns2)=O)CCC2(CCC(N(C)C(C3CC3F)=O)CC2)C1 N1(C(=O)CSCC2CCCO2)CC2(CCC2)CC1CNC(C1CCC=CCC1)=O C1(C(N2CCC(C(C)NC(CCCOCC)=O)CC2)=O)CC2(CCC2)CO1 c1(OC)ccc(Cl)c(CC(=O)NC2CC2NC(c2cc(OC)nn2C)=O)c1 C1(NC(=O)Cc2cnnn2C)CN(C(N)=O)CC1N(C)C.CC1C(=O)N1 C(CCC(C)NC(=O)C(C)C#N)NC(C1(CCCC)CC1)=O CN1N=C(CC(=O)NC2(C3CCCN3C(C3CCCN3C=O)=O)CC2)CC1=O C1(C(=O)NCCSCCC=C)CCCCN1C(c1ccncc1)=O.C(CN)N c1(CC)ccc(F)c(C(=O)N(CC(O)CNC(C2CCCC(C)(C)O2)=O)C)c1F C1(CC(=O)NCCN2CCOC2=O)COCCN1C(=O)COC1CC(F)(F)C1 C(=O)(C1=CCC(C)(C)CC1)NCC(C)=CC(=O)NC(C1CCCO1)C1CC1 CC1(C)CC(C(=O)NCC(C)(O)CNC(C2(C(F)F)CCCO2)=O)CC(C)(C)C1 N1(C(Cc2cc(C)ns2)=O)CCC2CC(C1)CN(C(=O)CC1CC1C1CC1)C2 CC1(NC(c2ccn(C3CCCC3)n2)=O)CCN(C(c2ncncc2Cl)=O)C1 C(=O)(C1=NOCC1)NC1CC(NC(c2c(OC(C)(C)C)scc2)=O)C1 CCCCCCC(=O)NCCOC1CN(C(c2cc(C)ccc2Cl)=O)C1 C1(NC(CCCc2ccc(C)s2)=O)C2CCN(C(=O)C(O)CC3CCOCC3)C12 CC1CC=C(C(=O)NCC2(F)CC(NC(c3nc4ccccc4[nH]3)=O)C2)CC1 C(C(C)(CCO)NC(c1ccc(CNC(=O)Cn2cc(CO)nn2)cn1)=O)OC C(CN=C(NCc1ncccc1O)NC1CCCC1)C1(C)COCCO1 C(=O)(C(F)(F)C(C)(C)O)NCC(C)(C)OCCNC(=O)CC1CC2CCC1O2 c1(C(N2C(CCC)CN(C(=O)C(CC(C)C)OC)CC2)=O)nc[nH]c2ncnc1-2 C(=O)(N=c1cc(Cl)nc(O)[nH]1)c1c(C(C)(C)C)nc(-c2ccccc2)[nH]1 c1(OC)cccc(OCC(N2CCC(CNC(=O)C=Cc3cccs3)C2)=O)c1 c1(C(N2CCOCC(NC(c3c(C)nco3)=O)C2)=O)ccc(C)c2ncccc12 c1(C(=O)NCc2cn(CC(CC)O)nn2)ccc(C2CCC23CCC3)cc1 C1(CC(=O)N(C(C)C(=O)NC)C)CCCN1C(=O)C=CC=C(Cl)Cl.CC(=O)N CCC(C)(COC)C(=O)N1CC(CC(F)C(=O)Nc2cncnc2O)C1 O=S1(=O)CC2CN(Cc3ncc(-c4cncc(F)c4)cc3Cl)CCN2C1 c1(CC(NOCC(N2CCC(CCC)C2)=O)=O)ccc(O)nn1 C1(C(C)NC(=O)NC2(c3ccccc3F)CCC2)CN(C(=O)OC(C)(C)C)CCO1 c1(C(=O)NCCN(C2CCCC2)C(C2CC3(CCCO3)C2)=O)cnn2c1CCC2 c1(NC(C2N(C(CC)=O)CC(F)C2)=O)ccc(O)cc1C(F)(F)F N1(Cc2n(CCC)ncn2)CC(N2CCN(C(=O)OC(C)(C)C)CC2)C(C)C1 N1(CC(=O)NC2C3(CN(C(COC)=O)C3)SCC2)C(=O)CC(C)(C)C1=O CCCCC(C(=O)NCC1C=CC(NC(=O)OC(C)(C)C)C1)NC(N)=O S(=O)(=O)(c1ccc(NCCC(=O)NC(C)(C)C)cc1Br)NC1C(OC)C(C)(C)C1 C1(OC)CCN(CCC(N2CCCCCC2c2ccccc2)=O)CC1C(=O)O C12(CNC(CCNS(CC)(=O)=O)=O)CC(CN1C(c1ccnn1CC#N)=O)C2 C1(NC(COCCC(C)C)=O)CCC2(CCCN(C(=O)CC(F)(F)C(C)C)C2)C1 C(=O)(C(C)(C)CCCC(=O)N1CCC(NC(=O)CC(F)(F)C(C)(F)F)C1)OC C1(C)(C(N(CCCCCNC(C2(CC)CC2)=O)C)=O)CCSCC1 CN1N=CC(CC(N2CC(O)(CCNC(=O)Cn3ccnn3)C2)=O)C1=O C(=O)(C1=Cc2cc(F)ccc2OC1)N(CC(C)NC(C(CC)C(C)O)=O)C Cc1onc(CC(N2CCCC2(C)CNC(=O)CSCC(C)C)=O)c1C#N C1(C)(C(N(CCC(=O)NCC(c2nncn2C)C)C2CC2)=O)CCOCC1 C1(C(=O)NCC(N2C(CC)CCC2)=O)CCN(c2ncccn2)C1.C(CC#N)S C12(C(=O)NC(C3OCC(C)OC3)C)CCC(NC(C3CN4CCC3CC4)=O)(CO1)C2 CC1CN(C(C2CCN2C)=O)CC1NC(C1(CN(C)C)CCCC1)=O CCC(CC)C(F)C(=O)NC(CC(=O)N(CCOC)CC)C(F)(F)F c1(NCC(COC)C)nccc(=NCC(OC)c2ccccc2)[nH]1 N1(c2ccc(NC(=O)NCC)cc2C(=O)OC)CC(C(F)(F)F)C(C)CC1C C1(C)(CNC(C(c2scc(C)n2)(F)F)=O)CN(C(C2CCCCC2)=O)C(C)(C)C1 Cc1nc(C(=O)N(CC(O)CNC(c2c[nH]c(=N)s2)=O)C)sc1C c1(CNC(=O)NC2CCCNC2C2CC2)ccc2c(c1)CC(=O)NC2 CCC(C)CC(=O)NC1CCCC1CNC(c1cn(C2CCOC2)nc1C)=O Cn1ccc(C=CC(=O)NCCOCC(=O)NCC(C)(C)CCO)c1 c1(C(=O)OC)n[nH]c2c(C(=O)N(C(C)CNC(c3cc(Cl)c[nH]3)=O)C)cccc12 c1(OC)ccc(F)c(OC2CCN(C3CC3)C2=O)c1.C12(CCC1)C(=O)NC2.COC C1(C(N(CCOCCN(C(=O)CNC=O)C)C)=O)CCCC2(CC2)C1 C1(NC(c2c(SC)cc(C)cc2)=O)CC2CCC(C1)N2C(=O)C(C)CCN(C)C N1(C(=O)Cc2cc(F)c(Cl)cc2Br)CC2CC(C2)c2ccc(Br)cc21 N1(C(c2n(C(C)C)ccn2)=O)CCC2CCC12CNC(=O)CCCCC#N Cc1cc(C=CC(=O)NC2(N3CCNC3=O)CC2)ccc1Br c1(C(=O)NC(CNC(c2c(CSC)cccn2)=O)C2CCC2)cc(Cl)ccc1O Cc1ccc(C(N2CCCC2CNC(c2ccsc2C(F)F)=O)=O)c(C2CC2)n1 c12cccc(c1)NC(=O)NC21CCC1.c1(CN(C(=O)OC)C)nnnn1CCO N1(C(C(C(CC)C)OC)=O)CC(O)(C2(CNC(=O)CCC3CC3)CC2)C1 C1(NC(C(C)OCCN(C)C)=O)CC(O)C(O)CC1C(=O)NCCOCCO C1(C(=O)NC(CNC(c2nc(C(=O)OC)oc2)=O)C2CC2)CCC(CO)CC1 Cc1ccc(CC(N2CCN(C(C3CCCCCC3)=O)C3CC23)=O)cc1[N+](=O)[O-] c1(CC)ccccc1C(=O)NC1(C)CCCC1NC(C1CC=CCO1)=O Cc1nn(C)cc1C(=O)NCC(C)(C)CNC(=O)C(F)CC1CCOC1 N1(C(=O)CN2CCC(F)CC2)CCCC2C1CCN2C(C1CCCCS1)=O CN1CCC(OCC(N2CC(O)CC2CNC(c2cccc(CO)n2)=O)=O)CC1 Nc1cc(C(=O)NC2CCC(CNC(C3CCCC34CC4)=O)CC2)ccc1Cl N1(C(CCCOC)=O)CC2(CC2)CC1CC(=O)Nc1cnc(O)c(F)c1 C1(CCNC(C2CCNC2=O)=O)CCCN(C(c2cncc(F)c2)=O)C1 C1(NC(c2c(OCC)nccc2)=O)CN(C(c2cocn2)=O)C2(CCCC2)C1 N1(CC)CC(NC(C2(CNC(=O)C(=O)N(C)C)CCCO2)=O)C(C)C1 c1(C(N2CC(C)C(NC(C3(S(N)(=O)=O)CCC3)=O)C2)=O)ccc2ccccc2n1 N1(C(CCOCCCNC(c2cc(C)c(=N)[nH]c2)=O)=O)CC(C)OC(C)(C)C1 C1(F)(CN(C(=O)Cc2cccnc2)C)CCCN(C(=O)C(C)(C2CC2)C2CC2)C1 c1(C(N2CCC(C)(CNC(CC=C=C)=O)C2)=O)ncc(N)cc1Cl C1(CC(C)NC(C=NOC)=O)CCN(C(c2ncccc2C(=O)OC(C)C)=O)CC1 CCC(CCC(=O)N1CCC(C)(CCO)CC1)NC(c1csc(SC)n1)=O c1(CN=c2scc(-c3c(C)nn(C)c3)[nH]2)c(F)ccc(Cl)c1Br C(=O)(CC1COc2ccccc21)NCCC1(O)CCCN(C(C(C=C)(C)C)=O)C1 c1(CC(C)C(=O)NCC2(C(=O)NCc3c[nH]c(=O)cn3)CCC2)ccccc1Cl CS(=O)c1ccc(CC(=O)NCCC2CC(NC(=O)C3=COCCO3)C2)cc1 c1(OC)cc(OC(F)(F)F)ccc1CNC(c1cc(-c2cnn(CC)c2)cs1)=O Cc1cc(C(=O)NCC(CNC(c2csc(Cl)c2)=O)C(F)(F)F)ncc1C#N CC1CCCC1(C(=O)NCC1NC(=O)NC1=O)NC(c1cnc(N)cn1)=O CC1CCN(C(c2cc(Cl)ns2)=O)CC1CNC(c1ccns1)=O C1(CNC(c2cnn(C)c2F)=O)CC2CCC1N2C(=O)C(C1CCCCC1)F N1(C(C2(NC(C)=O)CCSC2)=O)C2CCC(C2)C1C(N1CCN(C(C)C)CC1)=O c1(C(N2CCC(C)C(NC(=O)COC3CC3)C2)=O)cc(C#N)c(F)cc1F N1(C(C(CCOC)OC)=O)CC(NC(c2cc(C)ncc2C)=O)CCC1C C#CCC(C)(C)C(=O)NCC1CC(C)N(C(C2(c3cc(C)on3)CCC2)=O)C1 N1(CC(=O)NCC(CNC(c2c(CC)c(C)sc2)=O)O)C(=O)CC(C)(C)C1=O C1(C2(C)CC2)(OCC)CN(C=O)C1.C12CC(F)(C1)C(=O)NCC2=O.C1(C)CC1C.OC C12(C(N(CCNC(C(C)OCC(F)(F)F)=O)C)=O)COCC1C2 c12cn(nn1)C(C)C(=O)NC2.N1(CCSCCCC)CCOCC1 c1(NC(CSC)Cc2cccs2)cc(=O)n(C(C)C)nc1Cl CC(=O)CCCC(=O)N1CCC(CCF)(C(=O)N(C2CC(C(N)=O)C2)C)C1 C(=O)(C(CCO)N(C)C)NC(CCOC)CNC(c1ncsc1Br)=O C(=O)(CC(C)CC(C)C)N1CC(CNC(C(C2CCCC2)OCC)=O)C(C)CC1 C(=O)(CC(C)P(C)(C)=O)NC1(CCNC(C2CC(C)=C(C)CC2)=O)CCCC1 C(CCC(=O)NCc1csc(C(=O)NCCOC(C)C)c1)=C(C)C c1(NC(CNCC(=O)Nc2cc(Cl)sc2Cl)=O)cnc(F)cc1C(=O)NCCO C1(NC(c2nnnn2C(C)(C)CC)CCC)CCN(c2nccn2C)C1 c1(C(=O)NCC2CN(C(c3cc(C)c(C)[nH]3)=O)C(C)C2)c(C)nc(C)n1O C(c1ccc(F)cc1)=CC(=O)NC(CNC(c1cnn(CC)n1)=O)CC(C)C N(C1CN(C(=O)CCCC2CC2)Cc2ccccc21)C(C(C1CC1)OCC)=O Cc1cc(NC(=O)C(C)NC(=O)N(C)C)c[nH]1.C1(C(=O)NOC(F)F)(CC)CC1 N1(C(C2(C3CCCO3)CCCC2)=O)CCCCC1CNCc1ccc(F)nc1 N1(C(C(CC)c2ccccc2)=O)CC2CCN(C(=O)CCC(=O)OC)CC12 c1(C(=O)NCC(CC)NC(C2COC2)=O)ccc(Br)cc1Cl c1(C(N2CCCN(C(C(CCC)(C)C)=O)CCC2)=O)ccc2nc(=N)[nH]n2c1 C1(C(=O)NCCN(C(C2C3CCC23)=O)C2CC2)(CC)CCCCC1 C1(C(=O)NC(C)(C#N)c2ccccc2)C2CCC(C2)N1C(c1cccc(F)n1)=O C1(CNC(c2ccc(OC)cn2)=O)CC2(CCN(C(C3CCCO3)=O)CC2)CO1 c1(C(C)C)cc(C(=O)NC23CC(NC(=O)CC#N)(C2)C3)n[nH]1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(C)c2ccsc2)ccc(Cl)c(F)c1 C=C=C(C)CC(=O)N1CC2CC2(NC(c2sc(=N)[nH]c2C)=O)C1 c1(CC)nc(C)cc(=NC2CCC(C(=O)NC)C2)[nH]1 c1(C(=O)NC2CCC(C)N(C(=O)CSc3cn[nH]c3)C2)cnc2cc[nH]c2c1 CCCCCCCCNC(=O)C(=O)NCCN(C(C1CC1(C)CC)=O)CC1CC1 C1(C(=O)NCC(c2ncc[nH]2)C)CSCN1C(=O)C(O)CC1CCCC1 Cc1c(F)ccc(C(=O)NC2CCN(C(c3nc(=O)n(C)[nH]3)=O)C2C)c1C C=CC1(NC(c2ccn3ccsc23)=O)CCN(C(=O)OC(C)(C)C)C1 c1(C(N(CC(C)NC(C=CC=CC)=O)C)=O)cn(C(C)C)cc1C C1(C(=O)NC2CCCC(NC(C3CC(C)(O)C3)=O)C2)CNC(=O)CCC12CCC2 C(=O)(C(F)C(F)(F)F)NCC(CC)(C)NC(=O)C(=O)NCC1CC1 c1(N(C(C)(C)C)C(=O)OC(C2CC23CCOC3)=O)ccc(C2CCC2)cc1 C1(NC(=O)COc2ccc(Cl)cc2)CCN(Cc2nc(Cl)cs2)CC1F C1(C(=O)NCC(C)CNC(=O)Cc2ccon2)CC(=O)N(CC2CC2)C1 c1(C(=O)NCC(C)NC(c2ccc(OCC(F)(F)F)nn2)=O)ccc(CO)nc1 C12(C(=O)NCC(C)NC(C3(C4CCCCO4)CC3)=O)CCCN(CC1)C2 C1(CC(=O)NCC(C)OC)CC(NC(=O)CSc2cn[nH]c2)C1 N1(C(c2c(C#N)nc[nH]2)=O)CC2CC(NC(C3CCCO3)=O)CC2C1 C1(C(=O)Nc2cccc(CNC(CCC(=O)OC)=O)c2)CCS(=O)(=O)N1C N1(C(C2CC(CC)N(C(c3csc(C#N)c3)=O)CC2)=O)CCS(=O)C(C)C1 CC(C)C(CC(=O)N1CC(CNC(=O)C(C)O)C1)C(C)C Cc1nn(C)c(C)c1C(=O)NCC(C)CN(C(=O)C(C)Sc1ccc(Cl)cc1)C CC1CC(=O)NCC1C(=O)N(C1(C(=O)NCCC2CC(F)(F)C2)CCC1)C1CC1 C12(NC(c3csc(Cl)c3)=O)CCN(C(=O)CCCCc3ccccc3)CCC1C2 N(C1CCCc2n[nH]cc21)C(C(CC(C)(C)NC(CC(C)C(F)F)=O)F)=O c1(CC)cc(C(N2CCOCC2C2CCOC2)C(=O)NC(C)CC)cc(C)c1 C1(NC(c2sc(F)cc2Cl)=O)COCCN(C(=O)CCN2CCCCCC2)C1 c1(C(N2CC(C)C(NC(=O)CC3CC3)C2)=O)nn(C)c(=O)c2ccccc12 C1(N(C(c2c(C(C)C)noc2)=O)C)CC2CCC(C1)N2C(=O)C(C)n1cnnn1 N1(C(c2cnn(C(C)C)c2N)=O)CC(C)CN(C(=O)CCc2ncc[nH]2)CC1C C(=O)(C1=NOC(C(=O)OCCOc2nccs2)C1)N1CC(N(CCC)CCC)C1 c1(CC(=O)NCC2(C)CCN(C(COC)=O)CC2)cccc2c(C)csc12 c1(C(=O)NC2CCN(C(c3[nH]c(CC)c(Cl)n3)=O)C2)nccc2ccn(C)c12 N1(C(C2(C)CCN(C(C(CC=C)NC(C)=O)=O)C2)=O)CC2CC3CC2C1C3 C1(C(N2CCCCC2CN(C(=O)CCC2(C#N)CCC2)C)=O)(CC)CCNC1=O c1(OC)ccccc1NC(=O)NCC(N1CC(NC(=O)C(Cl)=CCl)C2CC12)=O C=C1CC(CNC(=O)CC(=O)NCC)(NC(=O)Nc2cnc(C3CC3)[nH]2)C1 C1(Cn2cc(C3(C)CCOC3)nn2)CCN(C(c2nc(Cl)cs2)=O)CC1 c1(CN2CC(C(=O)Nc3c(C)cccc3F)SCC2)cc(F)c(F)cc1O C1(CNC(C2(CC=C)CC=CC2)=O)(CNC(C2CCCCO2)=O)CC(F)(F)C1 c1(OC)cccc(CNC(=O)C(c2ccsc2C)N(c2cccc(F)c2)C)c1 c1(SCC)ccccc1C(=O)NC1CCCCC1CNC(c1nc(O)c(C)s1)=O N1(C(c2cncn(C)c2=O)=O)CC(C)(CNC(C2CC2C#N)=O)CC1(C)C Cc1cc(C(=O)NC(C2CCN(C(=O)CSc3nccn3C)CC2)C)nc(O)n1 C1(NC(c2cc(CC(C)C)on2)=O)C(C)CN(C(C2C3CCC23)=O)CC1C Cn1ccc(CN(CC(=O)OCC2CC(=O)C2)C(C2CCC(=O)C2)=O)c1 C(=O)(N1CCCN1C)c1c(CC(C=C)C)cccc1 CC1(CC2N(C(=O)Nc3ncccn3)CC2)CC(CN2CCOCC2)C1 CN1CCC2(CC1)CN(C(C1C=CCCN1C(=O)CSCCC#N)=O)C2 C(=O)(C(C)(C)C(F)(F)F)N1CCN(C(C(c2ccccc2Cl)C)=O)C(CC#N)C1 C(=O)(CC1=NNC(=O)C1)NCCC1CCN(C(C23C(CN(C(C)=O)C2)C3)=O)CC1 c1(CC(=O)NCC(C)CN(C)C(C2CC(C)OC2C)=O)cccnc1Cl n1(CCC)cc(-c2cscc2CN(CC(C)C(C)C)C)cn1 N1(CCNC(C(C2CN(C(=O)CC3CCCC3)C2)OC)=O)CCNC1=O N1(C(c2c(CNC(CC3CCCC(C)C3)=O)noc2)=O)CCNC(=O)CC1 c1(C(=O)NC2C(CNC(C(CSC)O)=O)CCC2)cc2ccccc2cn1 C#CCC(CC#C)C(=O)N1CCC(C)(CNC(c2cc(C)oc2CC)=O)C1 C1(N(C(=O)Cc2ccccc2Cl)CC)CCN(C(=O)Cc2ccsc2C)CC1 Cc1ccc(N)c(C(=O)NC2C3CN(C(c4cc5n(n4)CCO5)=O)CC23)c1F C1(NC(CCc2n(C)c(S)nn2)=O)CN(C(=O)Cn2cccc2)C2(CCC2)C1 c1(C(=O)NC(C(C)NC(C(CC)n2ccnc2)=O)C)c(Cl)ccc(F)c1F CC1CN(C(c2cc(Cl)cn2C)=O)CC(C)N(C(=O)CN2CCC(CO)CC2)C1 N1(CC(N2CCC(N(CC#C)C(c3cnc(Cl)s3)=O)C2)=O)C(=O)CC(C)(C)C1=O O=C1CCC2CN(C(C3CC(=O)N(C(F)F)C3)=O)CC2N1 c12ccnc(c1)C(=O)NCCS2.C1(CCC)CC(NC(=O)C=CCOC)C1 S(=O)(=O)(c1ccc(NCCC2CCCC2)cc1Br)NC1CCC(CC#N)C1 CP(C)(=O)CN1CC(C(N2CCCC(CO)(NC(=O)Cc3cocn3)C2)=O)C1 c1(C(N(CC(=O)Nc2cncnc2)C)=O)ccc(C#N)cc1F CC(C)CCCCCNC(c1nnnn1C1CC(F)(F)C1)(C)C1CC1 c1(NCC(n2ccnc2)C)ncccc1S(=O)(=O)NC(CC1CCCC1)CO C1(NC(c2ccc(C#C)o2)=O)CC12CCN(C(C1(OC)CCCC1)=O)CC2 c1(C(=O)NC23CC(CNC(c4ncc(F)cn4)=O)(C2)C3)cnc2nccn2c1 c1(OC)cccnc1NC(C1CCN(C(=O)C(c2ccc(Br)cc2)O)C1)=O CN1CCN(C(C2CCC(O)CNC2)=O)CC1CNC(c1ccc(F)cc1)=O CCC(CC(=O)N1CC(O)(CCCC(F)Cn2cc(C3CCC3)nn2)C1)C(C)C Cc1cc(C(=O)NCC(C)N(C)C(c2cc[nH]c2)=O)cc(Br)c1C C(=O)(C1=CCS(=O)(=O)C1)N(C1CN(C(CC2CCCN(C)C2)=O)CC12CC2)C C1(NC(=O)C=Cc2cnc[nH]2)COC2(C1)CN(C(=O)COc1ccc(Cl)cc1)C2 c1(C(=O)NC2C(C)N(Cc3cc(F)ccc3Cl)CCC2)ccc2nccn2c1 c1(C(=O)NC2CC(N(C(C3C(CC)C3)=O)C)C2)cc(-c2cccs2)on1 c1(C(=O)NCC(=CC(=O)NC(COC)CO)C)csnc1C c1(CC)nn(C)cc1C(=O)NCC1CC1CC(=O)NCC(COC)OC C12(CNC(C(C)(CO)NC(c3cnc(C4CC4)o3)=O)=O)CCC(C1)C(=O)N2 N1(C(C2(C(=O)OC)CC2)=O)CCC(C)CC(C(N2CC3C(N)C3C2)=O)C1.CCOCC Cc1ncc(C(=O)NC(CCNC(C2CCCC23CCC3)=O)C(C)C)cc1C#N O=C(N=c1[nH]nc(O)s1)C1=NOC2(CCN(C(C3CCCCC3)=O)CC2)C1 C(=O)(C(C)(C)C(F)(F)F)NCC(CC(C)C)NC(C1CCn2nnnc2C1)=O CC1CCSCCN1C(C1CCN(C(c2cc(O)cc(=O)o2)=O)CC1O)=O N1(C(=O)OC(C)(C)C)CCN(C(C2CN3CCCC2C3)=O)CC1CC(F)F c1(CN(c2cccnc2)C)cn(-c2cccnc2)nc1-c1ccccc1 C1(C(N(CCCO)C(C)C)=O)CCN(C(=O)C(C)Cc2ccco2)C12CC2 Cc1ccc2cc(C(=O)NC(CC(=O)NCCCN3CCCC3C)=O)[nH]c2c1 N1(C(c2cnc(CC)s2)=O)CCN(C(=O)C(C)SC)CC1c1ccccc1OC Cc1cc(O)ncc1C(N1CCC(F)(C(=O)NC2COC3(CCC3)C2)C1)=O c1(CCC(=O)NCCC2CC(NC(C3C(C=C)CC3)=O)C2)ccc(SCC)cc1 CCCC(CCC)C(=O)NC1CC2CCC1(CNC(c1cc3n(n1)CCC3)=O)C2 c1(OC)nn(C)cc1C(=O)NC1CCCC1NC(c1cncc(N)c1)=O C1(NC(c2cc(=O)cc(Cl)[nH]2)=O)CCN(C(=O)Cc2ccsn2)CC(O)C1 C=C(C)CC(C)C(=O)N1CCC(N2CCN(C(c3sc(F)cc3C)=O)CC2)C1 C1(CNC(CC=C(C)C)=O)OCCC1C(=O)N(CCCc1ccco1)C C#CCCCCC(=O)N1CCC(CC=C)(C(=O)NC(c2ccsc2)C)C1 C(=O)(CC1C(=O)N1)OC.c1(CSCC(=O)NCCOC(C)(C)C)nc[nH]n1 c1(C(=O)NC2CCN(C(C(CC)C3CCOCC3)=O)CC2)cc(O)c(F)cc1N C1(C(C(=O)NCCCc2ccncc2)F)CCN(C(c2cccn2C2CC2)=O)C1 C1(C)(c2ccccc2)CC(F)(F)CN1C(=O)CN(CCCCC(C)O)C(=O)CO c1(CNC(C2(C(C)(C)C)CCCCC2)=O)nc(CNC(C2(C)CC2F)=O)cc(O)n1 c1(NC(C2C(CNC(C(CCC)C#N)=O)OCC2)=O)ccn2nccc2c1 CCC(C)(C(=O)N(CCCNC(=O)C(c1ccc(Cl)cc1)=O)CC1CC1)C(F)F c1(C(=O)N)cnc2n1CCC2.c1(C(N2C(CC)(CC)CC2)=O)cccc(CO)n1 C(c1ccc(F)nc1)=CC(N1C(C)CC(NC(=O)CCc2ccc(Cl)nc2)C1)=O N1(CCC(=O)NCCC(C)(C)Cc2ccccc2)Cc2ccccc2C1 Cc1cnc(NCc2cccc(NC(C3CCCC3)=O)c2)nc1 c1(C(=O)NC(c2cn(C)nn2)C(=O)N(CCC#C)CCO)cccnc1O C1(CC(N2CCCC(N(C)C)C2)=O)N(C(=O)C=CCN2CCCC2)CCC1(C)C C(=O)(C(C)(C)CC(=O)N1C(C)C2CC1C2NC(=O)CCc1cocn1)OC C12(C(=O)NC(C)C3CC3)C(NC(C3CCC3C#N)=O)C3CC1C2C3 N1(c2cc(NC(C)C)ncn2)CCC2(CC1)CC2C(N1CCC2CCCC2C1)=O C(=O)(C(C(C)O)NC(C1CC(C)(NC(C2CCCC(=O)C2)=O)C1)=O)OC O(NC(=O)C(CNC(=O)CN(C)C)NC(=O)C(C)C)C(c1ccccn1)C n1(CC)ccc(NC(=O)C(COCc2ccccc2)OC)n1.C1(=O)C=CCN1 c1(OC)ccc(-c2nc(-c3ncn(CC(C)C)n3)n(C(C)C)n2)cc1OC C1(NC(c2cc(C(F)F)[nH]n2)=O)CC12CCN(C(=O)Cc1ccc(Cl)cc1)CC2 C1(NC(=O)CC2CC23CC3)CC(CN(C(=O)CCCc2ccccc2)C)C(O)C1 N1(C(CC2(OCC)CC2)=O)CCc2ccccc2C(NC(c2ccn(C)n2)=O)C1 c1(C(N2C(CNC(C=C(C)C)=O)CCC2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(c2c(OC)cc(Br)cn2)=O)CCC2(CCCN2C(=O)C=C2CCC2)C1 N1(C(C(C)OCC#C)=O)CCCC(C)(C)C1C(=O)NC1(c2ncccn2)CC1 c1(C(=O)NCC(CO)NC(C2C(C)OCCC2)=O)ccc2c(c1)CCC2 c1(C(=O)NC2C(C)(C)CN(C(=O)C(O)P(C)(C)=O)CC2)cccc2cnccc12 c1(COC(C2CC(NC(=O)CO)C2)=O)cncc(F)c1 C1(NC(C2CC2(Cl)Cl)=O)CCOC12CCN(C(c1ccc(Cl)s1)=O)CC2 C(=O)(C(C)(C)C(C)(F)F)NCCCOCCNC(c1cc(C)cc(O)n1)=O C1(NC(CCCc2ccc(C)cc2)=O)CN(C(C2CC2CF)=O)CC2(CCC2)C1 CC1N(C(c2conc2C(C)NC(=O)C=Cc2ccsc2)=O)CCOC1(C)C C1(C(=O)NCCCC)CCC(CNC(=O)COC2CCCC2)C1 N1(C(c2ccc(C)cc2Cl)=O)C2CCC1CN(C(=O)Cc1occc1C)C2 c1(CC(=O)NCC2(OCC)CN(C(CS(CC)=O)=O)C2)ccc(Cl)c(C)c1 c1(OC)ccc(CC(=O)NCC2CCCCN2C(c2cccnn2)=O)c(OC)c1 c1(C(=O)NCC2C3CN(C(CCC(C)OCC)=O)CC32)c(F)ccc(OC)c1N C1(CNC(CCOC(C)=O)=O)CC2CN(C(C3CNC(=O)CC3C)=O)CC12 N1(C(CCN(C)CC)=O)CCCN(C(c2cc(N3CCCC3)ccn2)=O)CC1C c1(C(=O)NCC(C)(C)CNC(=O)C2=CCCOC2)c(C(F)F)nc2ccccn12 CCC(C)(C)C(=O)C(=O)N1CC(F)(F)CC1(C)CNC(=O)CCn1ccnc1C C1(NC(CCC2C(C)C2)=O)C2CC1CN(C(C1(O)CCOCC1)=O)C2 C(N=c1[nH]c(Cl)nc2c1SCC2)c1cn(C2CCN(C(=O)CS(=O)(=O)C3CC3)C2)nn1 C1(CCC(=O)OC)CN(C(C2CC3(CCC3)C2)C(=O)Nc2ccco2)CCO1 CC(C)(CF)C(=O)N1CCC(N2CCN(C(c3scnc3C3CC3)=O)CC2)C1 c1(C(N(C)CC2N(C(CC(C)F)=O)CCC2)=O)cnnc(O)c1 CS(=O)(=O)CCNCC(N1CCCC1CO)=O N1(C(CCNC(COC)=O)=O)CC2CC2(NC(c2csc(CCC(F)(F)F)n2)=O)C1 C1(C2CCN(C(=O)C(C)CC3CCC3)C2)(NC(C=CC(C)C)=O)CC1 C1(NC(=O)C2CC2)CC2(CCN(C(C3C(C4CC4)C3(F)F)=O)CC2)C1 Cc1cc(N2CCN(CCNC(=O)Nc3csc(C)c3)CC2)nc(C(C)(C)C)n1 c1(C(N2CCN(C3CCN(C(C(C)(C)O)=O)C3)CC2)=O)ccc(NCCO)cc1 c1(OC)ccc(-n2cc(CNC(=O)C(C)NC(C3(C4(C)CC4)CC3)=O)nn2)cc1 Cc1nc(-c2ccccc2)oc1NC(=O)C(=O)NC(C1CCCC1)C#N c1(C(C(N(C(=O)COCc2nc(CC)no2)CC)C)C)csc(-c2cccs2)n1 c1(-c2nc(C(C3CC3)OC)nn2C2C(C)CCCC2C)cc2cnccc2[nH]1 C=CCC(C)(C)C(=O)NCCOC1CCN(C(=O)C(n2ccc(C)n2)C)C1 C12(Nc3cc(CC)ncn3)CCCC1CN(C(=O)CNS(=O)(=O)CC)C2 C(=O)(C1CCCc2cccnc21)NC1CCC(CNC(C(CC)=CC)=O)CC1 C#Cc1cn(C)nc1C(N1CCCC(C(=O)NCCC#CCC)CC1)=O CC1(C)CC2CC(C)(CN2C(=O)N=c2cc3n([nH]2)CCCN3)C1 c12cncc(c1)CN2.C1(C)(C(=O)OC)CC(C(=O)NC(C2CN(C(C)C)C2)=O)C1 N1(C(CSCCOC)=O)CC(NC(c2nccn3nccc23)=O)CC2(CCC2)C1 Cc1cc(C)n(CCC(N2CC(N(C)C(c3cc(C4CC4)on3)=O)C(O)C2)=O)n1 Cc1oc(CC#N)cc1C(=O)COC(C1(CSc2cnn(C)c2)CCC1)=O C(CCCCCC(F)(F)F)NCC(=O)NCC(c1ccccc1)OC(C)C c1(C(=O)NCCC(C)(C)NC(=O)CSc2cccs2)cc2c(nc1O)CCOC2 C(C(C)C(=O)NC(C)(CNC(=O)C(F)=C1CCCC1)CC)N(CC)CC N1(c2c(OC)cnc(Cl)n2)CCC(F)(F)C(CNC(=O)C(=O)NC(C)C)C1 C(=O)(C(F)(F)c1cscn1)NCCN(C(=O)CC1CC(F)C1)CC c1(C(=O)NCC(CNC(C2(CC=C)CCC2)=O)F)ccc2c(c1)OCO2 c1(C(C(=O)NCCCC)N(C)CCC(F)(F)F)ccc(SC2CC2C)s1 CC(C)(CS(C)(=O)=O)C(=O)NCC1CCC1NC(c1ccnc2ncnn12)=O C1(NC(C(C)c2ccco2)=O)CC2(CCN(C(=O)CC(C)(C)F)CC2)C1 CCCC(CC)C(=O)NC(Cn1cncn1)C(=O)NCCCN1CCCC1=O C1(C(=O)Nc2c(CC)nn(C)c2)CCN(C(=O)CC2=CCN(C)CC2)O1 C1(NC(Cc2cc(OC)no2)=O)CCC2(CC1)CN(C(C1CC1CF)=O)CCO2 CCCCCCCCCCC(=O)NC1(C)CCN(C(C2CC2(F)Cl)=O)CC1 N#Cc1cnc(NC(C2CC3CC3N2C(c2c(Cl)cccc2Br)=O)=O)c(Cl)c1 N1(C(c2ccc(OC)cc2)=O)CCC2(CCN(C(=O)C(CC)CC(F)(F)F)C2)C1 c1(NC(C2CC3N(C(CNC(N)=O)=O)C(CC3)C2)=O)ccc(Br)c([N+](=O)[O-])c1 c1(CN(C)CC2(C(=O)OC3CCC(C#N)C3)CCCC2)cccc(Br)c1 c1(-c2n(CC)nc(-c3ccccc3Cl)n2)cc(C)n2ncc(Br)c2n1 C1(C)(C(N(C)CC2CCCN(C)C2)=O)CC12CCN(C(c1cnccn1)=O)CC2 C1(NC(N2CC(C(=O)OC)OCC2)=O)CCCC12CC1(CC2)OCCO1 N1(C(COCC=C)=O)CCCC(C)C1CNC(=O)CCc1cn(C)nn1 c1(C(=O)NCC2CCCN(C(C(CCSC)O)=O)CC2)n[nH]c2c1CCSC2 C1(CNC(CC2C(C)=NOC2=O)=O)CN(C(=O)CCOC2COC2)CCC1(C)C c1(CC(=O)NCC(C2CCCC2)NC(C=C(C)C(C)C)=O)ccccn1 N1(C(c2cc(OCC)no2)=O)CCN(C(=O)CC2CC(OC)C2)CC1CF C1(CNC(C(CN(C)C)(C)C)=O)CCC(C)(C)CN1C(C1CCCCC1O)=O CC(C)C(C(=O)N1CCCC1c1ccc(N)cc1)n1nncn1.C1CCCC1 C1(NC(C(CCC)OCC)=O)CCC2CC1CN2C(c1nnc(CC)s1)=O c1(CNC(C2C(C(C)C)C2)=O)ccc2c(c1)CCCC2NC(=O)CC(C)(C)CF N1(C(C2CCCC23CCC3)=O)CC2CN(CCC3CCOC3)CC2C1 N1(C(CN(CC(C)(C)C)C)=O)CC=CC(NC(=O)C(O)C(F)F)C1 Cc1ccc(F)c(S(=O)(=O)N2CC3CCC(C2)C3C(=O)Nc2cc(F)ccn2)c1 N1(C(c2oc(CC)c(C)c2)=O)CCN(C(=O)C(c2cccnc2)=O)CCC1C CN(Cc1ccc(C#N)c(Cl)c1)N1CC(O)C2(CCCC2)C1 c1(C(=O)NC(CC2CN(C(C(=O)NCC)=O)C2)C)cnc(CC2CC2)nc1 C1(NC(Cc2scc(C)n2)=O)CCCC12CN(C(=O)Cc1cncs1)C2 Cn1nc(C2CC2)cc1CC(=O)NC1COCC1NC(c1coc(C(N)=O)c1)=O c1(C(=O)NCC2(NC(=O)C3CC3)CCCC2)ccc(F)c(CO)c1.CO N1(C(C2=CCCCC2C)=O)CCOC2(C1)CN(C(c1cnc(S)[nH]1)=O)C2 CC1(C)OCCOC1CC(=O)NC1CC(F)CN(C(=O)C2=CCCC2)C1 c1(OC)cc(CC(=O)NCCC(C)N(C(=O)C(C)NC(=O)C(C)(C)C)C)ccn1 c1(C(N2CCC(NC(C(Cc3ccccc3)NC(C)=O)=O)C2)=O)cnc(=N)[nH]c1 C1(CNC(C2CCC2)=O)CN(C(=O)CC2CC3(CC3)C2)CC(C(F)(F)F)O1 c1(OC)ccc(C(O)C(C)N(C(=O)C=CC=C(C)C)C2CC2)cc1 N1(C(c2c(CC)c[nH]c2)=O)CC2CCCC(CNC(C3CCCOCC3)=O)(C2)C1 CS(=O)(=O)CCC(=O)N1CC2C(CNC(=O)COc3cc(F)cc(F)c3)C2C1 N1(C(C(CC)=CCCC)=O)CC(N(C(=O)CC=C(Cl)Cl)C)C(C)(C)C1 c1(COC)nc(C(=O)NC(C)(C(=O)N(CCC(C)O)C)C2CCC2)co1 N1(C(C2(CC)CCC2)=O)CCN(C(C2OCCCC2(C)C)=O)CC(C)C1 C(=O)(CCC(=O)NN(C)C)NCC(CC(=O)N(CC(=O)OC)C)O CC(C)CC(CN=c1nc(N2CC3CCC(C2)O3)c2ncn(C)c2[nH]1)N(C)C c1(C(=O)NC2CCC(CNC(CSCCCC)=O)C2)cc2c(C)n[nH]c2cn1 C(CC(N)=O)(C(=O)NCCC1NC(=O)NC1=O)NC(C1(C)C(C)C1)=O CCCC(C)(O)C(=O)NC1C2CN(C(=O)CC3(n4cncn4)CC3)CC12 C1(OC)CCC(C)(CNC(=NCC2CC2)NC2CCN(C(C)=O)C2)CC1 Cc1onc(C2CC2)c1C(N1CCN(CC2CN(C(=O)C(=O)N(C)C)C2)CC1)=O N1(C(C(C(=O)OC)OC)=O)CCn2ncc(CNC(c3ccccc3)=O)c2C1 C1(OC)CN(C(=O)C(C)C(C)OC)CC1COC.C(=O)(CCCOCCOC)N CC(C)CC(CC(=O)NC1CC1c1cc[nH]n1)NC(=O)C(C)(O)C1CCC1 Cc1cc(Cl)ccc1CC(=O)NC1CN(C(C2(O)CCCCC2)=O)CCC1O C(=O)(C(F)(CNC(=O)CC(C)(C)C)C(C)C)N1CC(=C)C1 CCC(C)(C)C(C)CC(=O)N1CCC(CCCNC(=O)CP(C)(C)=O)CC1 Cc1cc(C=CC(N2CCC(CC(=O)NOCCN(C)C)C2)=O)on1 C1(C2CCN(C)CC2)(C(N(CC(CN(C(=O)Cc2ccon2)C)O)C)=O)CC1 N#Cc1ccc2oc(C(=O)NCc3ccnn3C3CCCCC3)cc2c1 C(=O)(CS(=O)CCC(F)(F)F)NCC(CNC(c1nccc(CC)c1)=O)O C1(C(C)NC(C2(C#C)CCC2)=O)CCCN(C(c2cscc2CCC)=O)C1 C1(C(N2CC(OC)C2)=O)CC2CC1CN(C(C1CC(F)(CF)C1)=O)C2 C=C(C)c1cc(C#N)ccc1NC(=O)NC(C)Cc1cc(C)cc(F)c1 Cc1cc(F)c(NC(c2sccc2NCC2CC2)=O)cc1F C1(F)(CNC(CCSCC)=O)CCN(CCCCNC(=O)C=CC2(C)COC2)C1 N1(C(CCC=C(C)C)=O)CCC(F)(CNC(c2cc(-c3ccncc3)[nH]n2)=O)C1 N1(Cc2c(C#N)cncc2)CC2CC(NC(c3cc(C(F)F)no3)=O)CC2C1 Cc1cccc2c1CCNC2C(=O)NCc1ccc(S(N)(=O)=O)nc1 N1(C(c2c(CC)cco2)=O)CCCCC(CNC(=O)CC2OCCO2)C1 C(CCN=[N+]=[N-])CC(=O)N(CC(C)O)CCNC(C(c1cccnc1)OC)=O c1(C(=O)NC(C2CN(Cc3ccc(C(=O)NC)cc3)C2)C)cc(Br)c(F)cc1F C=C1CC(C(=O)NC(c2ccc(C)s2)C)(CNC(=O)Cc2ccn(C)c2)C1 Cc1cnnc(O)c1C(=O)NCc1c[nH]nc1C(N1CCSC(C)C1)=O N1(C(C2N(C)CC(F)C2)=O)CCCC(O)(CNC(=O)Cc2ccon2)CC1 C1(NC(c2cnoc2C2CC2)=O)CCN(C(=O)Cc2ccc(O)nc2)CC1CO C(CN=c1[nH]ccc(=NCC2(C)CCCC2O)[nH]1)c1nnc(C)s1 C(CC(O)C(=O)NCC1(CC)C2=CC2=NO1)NC(C1CCCOCC1)=O C(=O)(C(O)Cn1cncn1)NCC(N1CC(SC)C1)=O CCCCCC(CC)C(=O)N(C(C)CCNC(c1nn(C)cc1N)=O)C C1(C(=O)NC(CC(C)C)CNC(c2c[nH]nc2Cl)=O)CCCCC12CC2 C1(C(=O)NCC2CCC(C)C2)CCCCN1C(C1(O)CCSCC1)=O C1(C(N2CCC(C)(F)CC2)=O)CC2CCCC2N1C(c1n[nH]c(=N)[nH]1)=O N1(C(c2ncc(OCC)nc2)=O)CCCC(NC(C2CC(C)N(CC)C2)=O)C1C Fc1c(N2CCN(Cc3ccc(F)c(Cl)c3)CC2)ccnc1Br c1(C(N2C(CNC(C3CC34CC4)=O)CCC2)=O)cc2ccccc2cn1 N1(C(CCCN(C(=O)OC)C)=O)CCC(CNC(c2ncsc2C)=O)C12CC2 N1(C(c2c(CC)scn2)=O)CCCCC1C(C)NC(=O)CCc1cccc(O)n1 C1(NC(c2n(C)cnc2)=O)CCN(C(=O)CC2CN3CCC2CC3)CC1O C1(NC(c2ccc[nH]2)=O)COCCC1NC(C1(C(=O)NC2C(CF)C2)CCC1)=O C1(NC(C=CC(CC)C)=O)CCC2(CC1)CN(C(=O)C(O)c1cnc[nH]1)CCO2 Cc1cc2c(cc1C)OC(C(N1CCC(CNC(=O)C(F)(F)CO)CC1)=O)C2 C1(NC(C2CCC23CCC3)=O)CCCCN(C(=O)CSc2ccc(Br)cc2)C1 C(CCCOC)(C(=O)NCCCF)CCCSC.C1(NCC)CCN(C)C1 c1(C(N(C2CCN(C(c3coc(C(F)F)c3)=O)CC2)C)=O)cc(O)cc(Cl)c1 C1(NC(C(CNC(Cc2cnc(C)s2)=O)C)=O)CCC(C2CC2)C1 O=C(N=c1[nH]nc2ccc(Cl)cn12)C1CCNC2(CCC2)C1 C1(C)(OCCC(=O)N(CCCNC(=O)CCCC2CCCC2)C)C(C)(C)C1(C)C C(C)(C1OCCc2sccc21)NC(=O)NC(c1ccccc1N(C)C)C c1(C(N2CCN(c3ccccc3C)CC2)C(=O)NCC)ccccc1C c1(C(=O)NC23C(CN(C(C(C=C)(C)CC)=O)C2)C3)ccc(Cl)c(C)c1Cl c1(C(N(CC(C)NC(=O)CC2CC2(C)C)C)=O)ccncc1F Cc1cccc(Cl)c1CC(=O)NC(C)CCCNC(=O)CC1CCCN1C C1(C(N2CCC(O)(CCNC(C3(F)CC3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1nc(F)ccc1N(C1CCNCCC1C)C(=O)C(F)F C(=O)(C(C)S(C)(=O)=O)N1CCC(C(C(N2C(CC)(CC)CC2)=O)C)CC1 N1(C(CN(C(C(CC)C(C)C)=O)C)=O)CCOC2COCC12 c1(-c2ccc(OC)c(O)c2)ccc2c(c1)CCN(C(c1cnc(Cl)cc1Cl)=O)C2 c1(C(N(CCCN(C)C(C2CCCC2(C)C)=O)C)=O)ccc2cncn2c1 CC1CN(C)CC1NC(c1conc1CNC(=O)C(C)CC1CC1)=O c1(CN2CCN(C(C(CCC)(C)C)=O)C(C)C2)cc(C#N)ccc1[N+](=O)[O-] C1(NC(CCCCNC(C23CCC(OC)C2C3)=O)=O)CC(C)N(C)CC1C c1(OC)nc(C)ncc1C(=O)NC1(CO)CCCN(C(C2(S(N)(=O)=O)CC2)=O)C1 S(=O)(=O)(c1ccc(NC(c2cc(OC)ccn2)C)cc1Br)NC(COC)COC N1(C(CC)C(=O)NC(C)Cc2ccc(Cl)cc2F)CCc2ccccc2C1 CCC(C)C(O)CNC(c1cccc(CSCc2cccnc2)c1)=O Cc1nc(SCC(=O)NCC(C)CNC(C2(O)CC2C(F)(F)F)=O)n[nH]1 Cn1ccc(NC(C2CC[Si](C)(C)C2)=O)c(O)c1=O C1(NC(C=NOC)=O)CC2CC(C1)N(C(=O)Cc1noc(C)c1C#N)C2 C1(OC)CCCC(Cc2nc(-c3ccccn3)nn2C2CCCCC2C)C1 c1(C(N2CCCC2Cn2cc(-c3ccco3)nn2)=O)cc(CO)n[nH]1 CCCC(CCC)CCCC(=O)N(CC)CC1CC1NC(=O)CN1CCSCC1 c1(ONC(C2(NC)CC2)=O)nc(C)no1.C1(NC(COC(C)=O)=O)CC(=C2CC2)C1 N1(Cc2nnc(C(C)(C)C)s2)CCS(=O)(=O)C(CCNC(C2(C)CC2CN)=O)C1 N1(C(C(=Cc2ccco2)C)=O)CCN(C(C23CSCC2C3)=O)C(CO)C1 C1(CN(C(=O)Cn2cnnn2)C2CC2)CCN(C(=O)CCn2ccccc2=O)CC1 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CCC(N=c2nc(C(C)C)[nH]s2)CC1 c1(C(N(CCNC(=O)C(CC)C2CCOCC2)CC)=O)ncc(Br)cc1C C(CCC(C)(C)NC(C1(CC(C)C)CC(=O)C1)=O)NC(C(C)OC)=O CCCC(C)(CC)C(=O)N1CC(CNC(=O)CCCC2CC2)(OC)C1 C1(C(N2C(C)(C)CCC2)=O)CCOCCN1C(C1CN2CCC1CC2)=O C1(NC(C2C3CC4C(C3)C24)=O)CCCN(C(c2ccnc(O)c2)=O)C1 c1(OCCCC(=O)NC2C(NC(c3c(C(C)C)c[nH]n3)=O)CC2)ccccc1Cl CCC(C)N=c1cc(C)[nH]c(=NCCCc2ncccc2Cl)[nH]1.n12ccnc1C2 C(C)(C)(CCC(=O)NC1CC(=O)N(C2CC2)C1)OC.c12ccn(c(=O)c1)[nH]c2=O C1(C)(C(NC(CCC2CCC(NC(C3CC(CCC)C3)=O)C2)=O)CC)CCCCO1 CC(C)(C)C(O)Cc1cn(C2(C(=O)O)CCN(C(=O)C3=NOCC3)C2)nn1 N1(C(C(c2c(C)cccc2)(C)C)=O)CCC(CNC(=O)C=C(Cl)Cl)C(F)(F)CC1 c1(-c2cn(CC(=O)N(CCCC3CC3C)CCOC)nn2)ccc(C(F)F)cc1 c1(C(N(C)CC2N(C(C3CCC(C)CC3)=O)CCC2)=O)nccc(N)c1Cl N1(C(c2c(CCC)nco2)=O)CCC(C(=O)N(C)Cc2ccns2)=C(F)C1 CC1CC(NC(c2cccnc2Cl)=O)CN1C(=O)CCCc1cncs1 C1(CCNC(c2cnc(C(C)C)o2)=O)CN(C(C2(CO)CC2)=O)CCCO1 CC(CCC(=O)NC(C)(C)C(=O)NC1CC1)NC(C1COCCN1C)=O c1(CCCNC(c2ccc(C(C)(C)C(F)(F)F)cc2)=O)ccc2c(c1)CCO2 c1(C(=O)OCC(C2CCC(NC(=O)OC(C)(C)C)CC2)(C)O)cc(F)ccc1O Cc1cncc(C(=O)NCC2CCCC(CNC(C3CN(C4COC4)C3)=O)C2)n1 C#CCCCC(C)C(=O)N1CC2(CCCC2)C1C(=O)NCCn1nncc1C C1(C(=O)NC(C)Cn2cc(CNC(C3(CSC)CC3)=O)nn2)CCCOCC1 N1(C(C2(C3N(C(c4nn(CC)c(C)c4)=O)CCC3)CC2)=O)CCC(O)C(O)C1 C1(CNC(CSc2cccc(C)c2)=O)C2CCC(C2)N1C(=O)COCC1CCC1 c1(OC)ccc(CCCC(=O)N2CC(NC(C3CC3(C)C(C)C)=O)C2)cc1 C=CCCC(C(=O)OC)NC(=O)CC(CC1CC1)NC(=O)C1=NOCC1 C(=O)(CCCC(C)(F)F)N1C2CC(CNC(c3ccc(C)nc3)=O)C1CC2 N1(CCC(=O)NCCCOC)CCC(C)C(NC(c2ccccc2OC)=O)C1 CC(C)C(F)(F)CC(=O)OCC1(C)CN(C2CN(C(=O)OC(C)(C)C)C2)C1=O Cc1ccc(F)cc1C1CC1C(N1CC(NC(=O)C2=NOC(C)C2)CC(O)C1)=O N1(C(C2CN(C(N(C)C)=O)C2)=O)CCCCC(NC(=O)CC2CCN(C)C2=O)C1 c1(C(=O)NCCC(C)NC(=O)CCSCC(N)=O)csc(-c2cnn(C)c2)n1 c1(OCC)cc2ccc(C(=O)NC3CNCC34CC4)cc2cn1 CCCCC(C)C(=O)N1CCN(C(=O)C(O)Cc2ccco2)C(CO)C1 CC(C)(C)C(=O)NCC(C1CCOC1)NC(c1cc(C(F)(F)F)n[nH]1)=O c1(C(=O)NCCC(C(=O)NCC(N)=O)OC)cccc(F)c1F C(CCC(C(=O)NCC1(C)CCC(C)CC1)NC(c1cc(Cl)cn1C)=O)OC C(=O)(CCCC(=O)N1CCC(NC(c2coc(Br)n2)=O)C(C)C1)NCCC CC(O)C(C(=O)N(CCCNC(C1CC1(C)C)=O)Cc1ccccc1)N(C)C C1(C(=O)NCC2CC(NC(C3=C(C)CCCC3)=O)C2)CCc2nnc(O)n2C1 CC(C)CC(C(=O)N1CCN(CCCNC(C2CC23CCC3)=O)CC1)C(C)C C1(C(C)C)CC2CCC(C1)N2C(=O)Nc1cnc(-c2cccs2)o1.N1(C)CC1 CCC(CC(=O)NC1CC2(C1)CC(CNC(=O)CN(S(=O)(=O)CC)C)C2)C(F)F N1(C(c2c(CC)nco2)=O)CCCC2C1CCCN2C(=O)CN1CCCCCC1 c1(SC)cc(C(=O)NCC2(NC(=O)CC3CC3(C)C)CC2)ccc1N n1(CC(=O)NCCCCC(C)NC(=O)CC23CCCC2C3)nc(O)ccc1=O c1(-c2onc(CC(=O)NC3C(=C)C3)n2)cc2c(cc1OC)OCO2 N1(C(c2ccccc2)C)CC23CCCC2(CNC3)C1 C1(C(=O)NC(CCC)CNC(C2CC(O)(C(F)(F)F)C2)=O)CN2CCN1CC2 C1(C(=O)NCCC(C)NC(Cn2c(C)ncc2)=O)CC12CCSCC2 c1(C2C(C(=O)NCCNC(C3(C(=O)NC(C)C)CCC3)=O)CC2)ccccc1Cl c1(C(=O)NCC(C)N(C)C(c2c[nH]nc2-c2ccccn2)=O)ccnn1C(F)F Cc1ccsc1CO.N1(C(CCSCCCC)=O)CCCC1C1CCCC1OC C1(C(N2CCN(CC(=O)NCc3c(C)cccc3)CC2)=O)CC(N)CCS1(=O)=O N1(C(C2(CCOC)CC2)=O)CCC(O)(CNC(=O)C=CC2(C)CCOCC2)C1 C(CC(C(=O)NC(c1cnc[nH]1)C)NC(c1cccc(CC)n1)=O)=CC CC(C)(O)C(F)C(=O)NC1CCC(C(=O)NOCC2(CCCO)CCCC2)C1 c1(N(CCOC)C)nc(=NCC2(c3ccccc3C#N)CC2)[nH]c2c1CSC2 c1(C(N2C(CNC(C3CC3F)=O)C=CC2)=O)nnn2c1CCCCC2 C1(N(C)C(C2CCNC(=O)C2)=O)CCC(NC(=O)CSCc2ccccc2)CC1 c1(CC)nn(C)c(CNC2CCN(CCC(F)(F)F)C2)c1Br c1(C(=O)NC2CC(NCc3ccc(F)s3)C2)ccc(CN(C)C)s1 c1(C(=O)NCC(CC)NC(c2c(N)cc(F)cc2F)=O)cnc2scc(C)n12 c1(C(=O)NC(c2cn(CC3CCOC3)nn2)C)sccc1F c1(OC)cc(C(=O)NC2CCN(C(=O)C=C(Cl)Cl)C(C)C2)cc([N+](=O)[O-])c1C c1(COC)nocc1C=O.c1(NC(c2cnsc2)=O)ccn(C(C)C)n1 N1(C(c2ccc(C(C)C)s2)=O)CCC2CCC(NC(C3(C)CC(C#N)C3)=O)C12 C1(C(=O)NC(C(C)NC(c2n[nH]c3c2CCOC3)=O)C)CC2OC(C)(C)OC2C1 CC(C)(C)C(C(=O)NCCCC1(NC(C2CC23CCOCC3)=O)CC1)NC(N)=O CC(C)(C)C(CNC(C1CC(=O)OC1(C)C)=O)C(=O)N1CCC1CF C=C(CC)CN=C(NCC1CC1(Cl)Cl)NC1CCN(c2ccc(F)cc2)C1 C1(C(=O)NCC2(O)CN(C(CCOCCOC)=O)C2)CC(C)OC(C)C1 C(CC1=CCCCCC1)NC(C=CC1N(C(CCCCC)=O)CCC1)=O C=CCCC(C(=O)NC1(C)CC(O)C1)NC(=O)C(OC)OC N1(C(=O)NCC2CCC3(CCC3)O2)CCCCC1C1CCCO1 C1(C(=O)NC(C#C)C(C)OC)CN(C(=O)CC2CC(=O)NC2=O)CC1C1CC1 C1(c2nnnn2Cc2ccccc2)(NC(CC)(CC)CCl)CC2CC1CC2(F)F C=Cc1cnn(C)c1C(=O)NCCOC(C)(C)CNC(c1cnccn1)=O S(=O)(=O)(c1cccc(OC(F)F)c1)N(C(CCC)C(=O)O)C1CC2CC1CN2 c1(NC(C2(C3N(C(C(C=C)OC)=O)CCC3)CC2)=O)cncc(F)c1 c1(C(N2C(CC(=O)NC(CC=C)C3CC3)COCC2)=O)ccc(F)c(F)c1 C(=O)(C(C)CC(F)(F)F)NCCOCC(N1CCC(CC)CC1)=O Cc1ccn(CC(=O)NCC2(CNC(c3cc(C(F)(F)F)n[nH]3)=O)CCC2)c(=O)c1 c1(CC)ccoc1C(=O)NC(C(=O)NCCN1CCC(O)C1)C1CCC1 Cc1cccc(C)c1OCC(=O)NCCC(O)C(F)(F)F C1(CC(=O)N(C)CC2(C)CCCO2)N(C(=O)CCP(C)(C)=O)CCC1(C)C C1(C(=O)NC(c2ncc(F)cc2F)C)CC(=O)N(C)C1c1ccc(Cl)c(Cl)c1 C(=O)(CCC(=O)NN(C)C)NC(C(=O)N1CCN(CC)CC1)CC(F)F c1(C(N2CC(CNC(c3ccc(C)[nH]3)=O)C(C)CC2)=O)c(C)cc(C)oc1=O C1(C(N(C(CC(=O)OC)C)C)=O)COC2(C1)CN(C(c1cc(O)ncn1)=O)C2 c1(C(N(C(C)C)CCN(C)C(C2CC(=O)C2(C)C)=O)=O)c2c(nn1C)CCCC2 C1(O)(CNC(CCc2cc(C)[nH]n2)=O)CCN(C(c2cnn(C3CC3)c2C)=O)C1 N1(C2CCC(C)CC2)C(=O)NC(c2cc3ncccn3n2)C2=C1C(C)CN(C)C2=O CCCCC(CC)C(=O)NC1C2CCC1N(C(c1cncc3ccsc13)=O)C2 Cc1ccc(F)c(-c2ccc(CN(C(c3sc(C)nc3C)=O)CCO)nc2)c1 c1(CC)cccc(S(=O)(=O)N2CCC(C#N)(NC(c3cccc(I)c3C)=O)C2)c1 C1(CNC(CN2C(C)CC2)=O)CN(C(C23CCCC(CO2)C3)=O)CCC12CCC2 N1(C(Cn2c(C)nc(C)n2)=O)CCCC(F)(CNC(=O)COC2CCCCC2)C1 c1(C(=O)NCC2C(CC)CN(C(=O)CC(C)(F)F)CC2)nc2ncccn2n1 c1(C(=O)NCC(CC(C)C)NC(CCCC(C)=O)=O)[nH]nc2c1COC2(C)C c1(CNC(=O)NCCNC(C2OCCC2F)=O)ccc(O)cc1F C=CCCN=C(NCCC(C(F)(F)F)OCC)NC1CCCN(C(=O)OCC)C1 N(C1CCCc2cc(CNC(c3cscc3C)=O)ccc21)C(C1CC(SC)C1)=O C(=O)(C(O)C1=CCCCC1)N1CCOCC(F)(CNC(=O)C2=COCCC2)C1 C1(CNC(N2CC3(COCC(C(=O)O)O3)C2)=O)CCc2nncn2CC1 C1(C(=O)NC2CC3(C(NC(C4CCSCC4)=O)C3)C2)Cc2c(F)cccc2O1 C1(NC(C2N(C(=O)NCc3n(C)ccn3)CCCC2)=O)COc2ccccc2C1 CC(C)(CC(F)F)C(=O)NCC1CC(NC(c2ccccc2C(F)F)=O)C1 c1(CC)ccc(C(=O)N(C2CCN(C(=O)CC34CCN3CCC4)C2)C)cc1 N1(CCN)CCCOC1=O.C12CCC1(C)CNC(=O)N(C)C2c1nccn1C CCCCCCC(C)CC(=O)N1CC(NC(c2cscc2Cl)=O)C1 CC(O)C(F)(F)C(=O)NC1(c2ccccc2)CCN(C(C2CCOC2=O)=O)CC1 CC(C)CC(C)(CNC(=O)C(C)(F)c1ccccc1)NC(=O)COC1CC1 n1(CC)cnnc1C(=O)NC1CCC(CNC(=O)CC2CNC(=O)O2)C1 c1(C(C)(C)C)ccccc1C(=O)NCC1CN(C(C2CC23CC(O)C3)=O)CCO1 C1(C(=O)NC2(CC)CN(C(CCCOCC)=O)C2)CCCCC1F c1(C(=O)NC2CC(CNC(C3(SC)CC3)=O)C2)ccc(C)o1 N1(C(CCCOC(C)C)=O)C2CC=C(C(=O)NCC(C)CCCC(C)C)C1CC2 c1(N2C(C3CCCN(C(C4CC(CF)C4)=O)C3)CCCC2)ccc([N+](=O)[O-])cn1 N1(Cc2c(C)nn(C)c2)CCC2(CCN(C(c3cnc(Br)s3)=O)C2)C1 C#Cc1ccccc1CC(N1CCN(C(C2CC3(C2)CC3F)=O)CC1COC)=O CCCCCC(C(=O)N1CCCC2(C1)CN(C(=O)CN(C)C1CC1)C2)C(C)C CCC(C)(C)C(C)CC(=O)N1CCCC1CNC(=O)C(=O)C(C)(C)C c1(OC)ccc(C)c(C(=O)NCC(F)CNC(=O)C(C)(O)Cc2ccccc2)c1 n1(Cc2cc(C(=O)NC3CC(CNC(=O)C(F)F)C3)[nH]n2)ccccc1=O c1(C(=O)NC(C2CCN(c3ccnc(OC)n3)C2)C)ccc2nc(CO)[nH]c2c1 C(CNC(=O)CC1(O)CCC1)(C(=O)N(CCC(N)=O)Cc1ccccc1)N(C)C c1(C(CC)NS(=O)(=O)CC2(OC)CCC2)cnn(C2CCC2)c1 C1(CC(=O)NC2(C3CN(C(C(C)CN(C)C)=O)C3)CC2)CC2(CCC2)CCO1 C1(NC(C(N2CCCC(C)C2)=O)=O)CCN(C(=O)CCc2cccnc2)C12CC2 N1(C(C(C(=O)OCC)OC)=O)CCC(C(=O)NC(C)CS(N)(=O)=O)C12CCC2 CCC(F)(F)CC(=O)NC(CC(N)=O)C(=O)N(C)CC1CCCC2CC12 Cc1nn(CC(N2CC(F)(CNC(c3cn[nH]c3)=O)C2)=O)cc1Cl c1(C(=O)NC2(CC=C)CN(C(=O)C(c3cnn(C)c3)=O)C2)cccn(O)c1=O C(=O)(C(=O)CCC(C)C)N(CCC(N1CCC(N(C)C)C(C)C1)=O)CC=C Cc1nc(C)c(C(=O)NCC(C)NC(=O)C(C)(F)c2ccon2)o1 c1(CCC(=O)Nc2ccccc2C(=O)O)ccc(F)c(F)c1 c1(C(N(CCC(=O)NCc2nc[nH]n2)CC#C)=O)cc(O)ncn1 N1(C(c2cncc(N3CCCC3)n2)=O)CCN(C(C2CC2(Cl)Cl)=O)C(C2CC2)C1 C(=O)(C1Cc2ccccc21)NC(C(C)NC(C(CC=C)CC=C)=O)(C)C c1(C(=O)NC(CC)CNC(c2cc(N)cnc2C)=O)cnc2n(c1=O)CCS2 C(=O)(C(CC1(CO)CCC1)NC(C)=O)OCC.C1(C(=O)N(CCS)C(C)C)CCCO1 N1(C(C2CC(OC)CN2C(=O)CC2CCCNC2=O)=O)CCC2CN(C)CC2C1 O=C(CCCC(F)(F)F)N1CC2CC(C1)C2NC(=O)C(F)(F)C1(O)CCCC1 C1(C(=O)NCC(CC=C)NC(=O)CCCN2CCCC2)CC(S(C)(=O)=O)C1 N1(C(c2cc(CC)no2)=O)CC2CC3CC2C1C3NC(=O)Cc1cccc(C)c1 N1(C(c2cc(CNC(C3(OC)CCCOC3)=O)ncc2)=O)CCCC2(CC2)C1 c1(-c2nc(CC(CC)(C)CC)on2)cccnc1N=[N+]=[N-] N1(C(COC(C)=O)=O)CCN(C(C2CNC(=O)C2)=O)C(C(C)C)C1 c1(C(=O)NCC2CN(C(C3CC(C4CCC4)C3)=O)CCO2)ccc2c(c1)OCO2 C1(O)(C(=O)OC)CCN(C(c2cnoc2NCc2csc(C(C)C)n2)=O)C1 C1(C(=O)NC2CN(C(C(CC)(F)F)=O)CC2O)Cc2ccccc2C1(C)C Cc1nc2ccccn2c1CC(=O)NCC1CCN(C(C2CC(F)C(=O)N2)=O)C1 N1(C(COCCOC)=O)CCC2(CC1)CC(C)N(C(c1cc([N+](=O)[O-])n[nH]1)=O)C2 C(c1cccnc1)=CCC(C1CC1)N.CC(CCCNC(=O)N)c1ccccc1 C1(C#N)(C(N2C(C(=O)NC(CCOC)COC)CCC2C(C)C)=O)CCCCC1 C1(C(c2ccccc2)OC)CN(S(=O)(=O)c2cc(Br)c(Br)s2)CC(C)(C)S1(=O)=O N1(C(CNC(=O)OC)=O)CCC(C2CN(C(c3cc(O)nc(O)n3)=O)C2)CC1 C1(CNC(C=CC=CC)=O)CN(C(c2cccc(CC(C)C)c2)=O)CCO1 Cn1ccc(=O)c(C(N2CCN(C3CCN(C(=O)C(F)C4CCC4)C3)CC2)=O)c1 N1(CCOCC)CC(NC(NC2CCCCC2)=O)CCC1C.c1(CO)ccsc1C c1(C(=O)NCC2N(C(C3CC(C)OC(C)C3)=O)CCCC2)cc(N)c(F)cc1F C#Cc1cccc(C(N2CC3CC2C3C(=O)Nc2cnn(C3CC3)c2C)=O)c1 C1(NC(C(C)(C)OCC)=O)CN(C(c2ccc(O)nn2)=O)CCC1O c1(C(=O)NC(C(=O)N2CCC(COC)C2)CCOCCO)cnn(C)c(=O)c1 c1(CC(N2C(CC)C(NC(=O)CN3CCC(F)CC3)CC2)=O)cc(F)cc(F)c1 N1(C(C(C)SCCCC)=O)CC2CC(C1)CN(C(=O)COCCSC)C2 CC(O)C(C(=O)NCC1CC1C(c1ccccc1)C)NC(c1cnn(C)n1)=O C(=O)(C(C)CCCC(C)C)NCC1N(C(C(n2c(C)ccn2)C)=O)CC(C)(C)C1 C=CCC(C(=O)NC(C)CCCO)NC(c1cnn(CCC)c1)=O c1(C(N2CCOCC2C2(C)CC2)C(=O)NCCOC)cc(OC)c(Br)c(OC)c1 C#Cc1cc(C(N2CC(NC(=O)CCC3CC3(F)F)C(CO)C2)=O)cc(F)c1 C1(CCNC(C2CC(CNC(C3(CC)CCO3)=O)C2)=O)CCCC2CC12 Cc1sc(Cl)nc1C(=O)NC(c1ccc(CNC(=O)C=Cc2ccsc2)cc1)C c1(C(N2CC(NC(C(CC)N(C)C)=O)C(C)C2)=O)cc(OC)cc(C(=O)OC)n1 c1(C(N2C(C)CC(CNC(C3(OCC)CCC3)=O)C2)=O)nn(C)c(C)c1Br CC(C)C(C)(O)C(=O)NC1CC2(C1)CC(CNC(=O)Cc1cc(Cl)ccc1Cl)C2 c1(NC(c2c(Cl)ccc(NC)c2)=O)cc2cc[nH]c2cc1F N1(CCNC(c2ccc[n+]([O-])c2)=O)CCCN(C(=O)C(F)CC2CCC2)CC1 C(=O)(C(F)C(CC)CC)N1C2CC(C(=O)NC(C#C)(C)C3CC3)C1CC2 C1(CNC(c2n(CC=C)ccc2)=O)CC(C)(C)CCC1NC(C1(C)CCC1)=O c1(CC)ccccc1CC(=O)OCC1CCCC1N(C(=O)Cc1ccsc1)CC CC1CN(C(=O)C=CCO)CC(C)N1C(C1CN(S(C)(=O)=O)C1)=O CC(C(=O)OC(C)(C)C)C(=O)NCC1CC(NC(c2cc(C(N)=O)n(C)n2)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)NC1CC(CNC(c2ocnc2C(F)F)=O)C1 C1(CC#C)CN(C(c2cnn(CN)c2)=O)C12CCC2 c1(Cc2scc(CNC3CC(CC)C3)n2)ccc(Cl)cc1 c1(CC(=O)NCC(CNC(c2c(C)ccnn2)=O)O)ccc(Br)cc1F CCCC(CNC(=O)C(C)n1ccnn1)C(=O)NCCC(C)(C)C C(=O)(C1CCc2cccnc21)NCCNC(CC(C)(O)c1ccccc1)=O C1(CCC2N(C(C(F)=CC)=O)CCC2)CCCCN1C(=O)Cn1cccn1 C1(F)(CNC(c2c(C)nn(C)n2)=O)CCN(C(c2cnn(CCO)c2C)=O)CC1 c1(N(CC(C)N(C(C)=O)C)C)ncnc(NCc2cc(-c3ccco3)on2)c1C c1(C(=O)NCCN(C2CCCC2)C(CN2C(C)CC2)=O)c(F)c(F)cc(F)c1F C#Cc1cnc(C(=O)N(CCCCCNC(C23CCOC(C)(C2)C3)=O)C)c(C)c1 CCCS(=O)(=O)CC(=O)NCC1CN(C(c2cnc(O)cc2OC)=O)CC1C C(C(F)(F)C(C)(C)C)NC1(c2nnnn2C2CC2)C(CC=C)OCC1 C1(NC(C(COC)O)=O)CN(C(=O)CC=Cc2ccc(F)cc2)CC12CC2 C(CCC(=O)N(CC(=O)NC(CC1CCCC1)CO)C1CC1)OCC CCC(F)(F)C(C)(C)C(=O)N1CCC(C2(NC(c3nc(C4CC4)cs3)=O)CC2)C1 C1(CNC(c2cnc(NC(C)=O)s2)=O)CN(C(c2ncc[nH]c2=O)=O)CC1(C)C c1(NC(c2cc(-n3ccnc3)ccn2)c2n(CC)nnn2)ccc(Cl)cc1C c1(SCC(=O)NC2C(NC(c3on(C)c(=O)c3)=O)CCC2)nc2ccccc2s1 C1(CNC(C(C)OC)=O)C(C)CCCN1C(c1sccc1C)=O Cc1cc(=O)c(C(N2CCOCC2CCNC(C2CC2(C)C)=O)=O)cn1C C=C1COc2c(C(N3CCC4(CC3)CC4CNC(=O)C=C3CCC3)=O)cnn2C1 C(=O)(N1NC(=O)CC12CCCCC2)c1noc(-c2ccccc2OC)c1C.CC CC(CCC(=O)N(CCCc1ccco1)C)NC(C1CC1(C)C(F)F)=O C=CCC(CC(=O)N(CC(F)(F)Cl)C)NC(=O)C(C)(C)C1CCOC1 C(=O)(C(=O)CC(C)CC)N(CC(N1CCCC(OCC#C)C1)=O)CCC C1(CNC(C=CC(CC)C)=O)CN(C(=O)CN2CCC(C)(C)C2)CC1(C)C N1(C(c2cccc(N(C)C)n2)=O)C(=O)CCC(Sc2ccccn2)C1=O C1(NC(=O)CC2CCSCC2)CN(C(c2cc(Cl)no2)=O)CC2CC12 C1(C(N2CCC(N(C(=O)CCN3CCC3)CC)C2)=O)Cc2cc(F)cc(F)c2O1 Cc1ccc(F)cc1C(N1CCC(C(C)NC(=O)CCCC(N)=O)C1)=O CN1CCC(CCNC(=O)CCN(C)C(C2CCCCC2)=O)C1=O CC1CN(C(=O)CC2CCSCC2)CCC1C(=O)N1CCCO1 C=CC(C)(C)CC(=O)NCCC1(NC(C2COCC(C)O2)=O)CCCC1 N1(C(C)C)CC(NC(=O)NCC2(Cc3ccccc3)CCCCC2)CC1=O CCC(CC(=O)N(C(C)C(=O)N1CCC1CC1CC1)C)C(C)(C)C c1(CC(=O)N(CC(O)CN(C(=O)CCCF)C)C)cc(Cl)n(C)n1 c1(CC(=O)NC2(CC)CCOC2)cc(F)cc2c1OCOC2 C(CC(F)F)(C(=O)N1CCC(N(C)CC)C1C)N(C(C(F)=CCC)=O)C C1(CNC(CC=C(C)C)=O)CCN(C(=O)CN2CCCC2=O)CC1C1CC1 C1(CC(=O)N(C(=O)C(CC2CCC2)OC2CCC2)C2C(C)C2C)OCCC1(C)C C12(CNC(=O)OC(C)(C)C)CC(C1)C(CSc1ccccc1)O2 C(CC1=CCCCCC1)NC(CC1C2CN(C(C3(CC)CCCO3)=O)CC21)=O c1(CN(CCNC(c2c[nH]c(=N)o2)=O)C(C23COCC2C3)=O)cccc(Cl)c1 C(=O)(CCC(=O)NC(C)CC(C)NC(C1(C)C=CCC1)=O)OC N1(C(C=C(CC)C)=O)CC(N2CCC2)C(CNC(=O)C(c2ccccn2)O)C1 Cc1cnc(C(=O)NCC2(CNC(=O)CCCN(C)C)CCC2)c(Br)c1 n1(CC(N2CCC(C)C2CNC(C2CCCC2)=O)=O)nc2ccccn2c1=O C1(NC(COCCOC)=O)CN(C(=O)Cn2cc(CO)nn2)CCC1CO C(=O)(C(CC)C(=O)N1CCC(F)(CNC(=O)CCc2ncccn2)CC1)OCC N1(C(C(C)(F)F)=O)CC2CN(C(c3ccc(F)cc3Br)=O)CC(C1)O2 C1(C)(CNC(c2cc(SC)oc2)=O)CCCN1c1nnc(CO)s1 c1(C(N2CC(OC)C(NC(=O)C3=CCCC3)C2)=O)nc[nH]c2ncnc1-2 c12cccc(c1)CNc1cc-2cs1.c1(CC(=O)O)cccc(Cn2ccnc2)n1 c1(CC)ccc(C(=O)NCCC(C)NC(=O)C(C)OCc2ccccc2)s1 c1(C(=O)Nc2nnc(CCSC)s2)cn(-c2ccccc2)nc1-c1ccccc1 N1(C(c2nn(CC)c(C)c2)=O)CCC2(CC2C(=O)Nc2cccc(C3CC3)n2)C1 CS(=O)(=O)c1sccc1C(N1CCC(CCNC(c2occc2Cl)=O)C1)=O Cc1nn(C)cc1-c1ccc(C(=O)NC(C)C(=O)Nc2ccccc2)s1 C=C(C)CC(C(=O)OC)NC(C1CCCCN1C(c1cnc(O)n1CC)=O)=O c1(CC)scnc1C(=O)NCCOCCCCN(C)C(C1CCC1CC)=O N#Cc1cc(C(=O)NCC2(O)CC(C(=O)NC(C)C3CC3)C2)c[nH]1 CCCC(CC)C(=O)NCC1CCN1C(c1ccc(OCC(F)F)cc1)=O c1(C(N2CC(NC(C3C(C)COCC3)=O)C2)=O)cn2ccc(Br)cc2n1 N1(C(CC2(OCC)CC2)=O)CCC(C(=O)N(C(COC)CC)C)(CC)C1 CN1C(=O)CC(C(N2CCCCC2CCNC(=O)C(F)(F)CO)=O)NC1=O CC(CN(C)C(C1CCC=CC1NC(c1cnnn1C)=O)=O)C(F)(F)F c1(C(=O)NCC2(O)CN(Cc3ccccc3)C2)ccc(I)cc1Br C1(C(=O)NC(C)Cn2cc(-c3cccnc3C(=O)O)nn2)CC2(C1)CC(F)(F)C2 C(CNC(c1cccc(F)c1)=O)(C(C)C(C)C)NC(c1ccc(COC)cn1)=O c1(C(N2CCC(C(C)NC(COC(CC)(C)C)=O)C2)=O)ccc2nc(O)oc2c1 CN1CCCCC1CC(=O)NCCCC1CCCCN1C(=O)Cn1cc(Cl)cn1 Cc1nc(C(=O)NCC2COC(CNC(c3c[nH]c(C(F)(F)F)c3)=O)C2)nn1C C1(CC=C)(NC(=O)Cc2nc[nH]n2)CCCN(C(=O)C=C2CCCCC2(C)C)C1 c1(OC)cc(C(=O)NCCCCN(C)C(c2cccn2C2CCCC2)=O)sn1 N1(C(C23CC(NC(C4C(COC)CC4)=O)(C2)C3)=O)CCCNC(=O)CC1 n1(C(C)C)cnc(C(=O)NCC(CO)NC(=O)C(C)(C)c2cccs2)n1 c1(NC(C=CCN(C(=O)CC2CCCC(O)C2)C)=O)cccn2nccc12 c1(OCC)ncc2ccc(NC(=O)Cc3ccnc(Cl)c3F)cc2n1 N1(C(c2cc(OC)n[nH]2)=O)CC(NC(=O)CCCOC(C)=O)CC12CCCCC2 Cc1cccc(C)c1N1CCN(C(c2c(C)ncn2C)C(=O)NC2CCC2)CC1 N1(C(C(C(C)C)(C)C)=O)CC23CCCCC2(C1)CN(C(c1cncc(F)c1)=O)C3 C1(C(N(c2cccc(O)c2)C)=O)Nc2ccccc2C1(C)C.C(C(F)(F)F)OCC#N N1(C(CN(C(C)C)C)=O)CCOC(C(=O)NCCc2cn(C)cn2)CC1 C12(CNC(C3(CC(C)C)CC3)=O)CC1CN(C(C1(O)CC(C(=O)O)C1)=O)C2 C1(NC(c2[nH]cc3c2CCC3)=O)CCN(C(=O)Cc2ccncc2)CC1F c1(CC(=O)N(c2ccc(OC)cc2Cl)C)cccc2ncccc12 c1(CC2CN(CC)C2)ccc(C(N2CCC(N(c3ccccc3)C)C2)=O)cn1 N1(C2C(NC(C3CCCCC34OCCO4)=O)CC(C)O2)CCC2(CCCCCC2)C1 c1(C(=O)NCC2C=CC(NC(C(C(C)C)NC=O)=O)C2)noc2ncccc12 c1(C(=O)NCCCOCCCNC(CC2(C)CCC2)=O)c[nH]cc1Br C1(C(=O)NC(CCOC)C)CC=CC(NC(=O)CC2CCOC2C)C1 C1(NC(C(C)OC)=O)CC2CC1N(C(C1CCN(OC)CC1)=O)C2 CC1C(NC(=O)C=CSc2nc[nH]n2)CCCN1C(=O)Cn1cnc([N+](=O)[O-])n1 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CC2NC(c1cccc2nccn12)=O Cc1c(I)nn(C)c1C(N1CCC(CN(C)C)C1)C(=O)Nc1ccccc1Cl CCCCC(CC)CC(=O)N1CCCC(NC(c2nn(CCC)cc2Cl)=O)C1C N1(C(C2CC(=C)C2)=O)CC(C)CN(C(c2nc(Cl)nnc2NC2CC2)=O)C(C)C1 C1(C(N2CCOCC2CC2CC2)=O)CCCCN1C(=O)C(C1CC1)C1CC1 c1(OC)ccc2c(C(=O)N(CC(C)N(C)C(c3ccc(C)n3C)=O)C)n[nH]c2c1 N1(C(CC2CC(OC)C2)=O)CCCC1C1(NC(C2(Cl)CC2(F)F)=O)CC1 C12CCCC(C1)CN(C(CNC(=O)CC1CC1)C1CC1)C2=O.N1(S(C)(=O)=O)CCCC1 C12(NC(CC=CC)=O)CCN(CC1)C2=O.C1(SC)CCN(C)C1C c1(C(=O)NCCNC(C2CC(C)(C)O2)=O)c(Cl)ccc(Br)c1F c1(OC)cccc(C(C(=O)NCC2CC3CC3N2C(=O)CCCC#N)OC)c1 Cc1oc2cc(C(=O)NC3CCN(C(=O)C(C)S(C)(=O)=O)C(C)C3)[nH]c2c1C CCC(C(=O)N(C1CCCN(C(c2ccc(C)cc2)=O)C1)CC1CC1)C(C)C C1(C(=O)NCC(CC)(C)NC(=O)CNC(c2nnc(C)s2)=O)CC2(CC2)CO1 N1(C(c2c(C)c[nH]c2)=O)CC2(NC(=O)C3Cc4ccccc43)CCCC2(F)C1 Cc1cc(C(N2CCN(C(c3ccc(CO)o3)=O)CC2)=O)c2c(c1)C(C)CCN2 c1(C(=O)NCCC(CNC(COCCC)=O)O)cc(C(C)C)cc(O)c1 CC1(CCO)CCCN1C(=O)C(C1CCN(C(c2ccnc(O)c2)=O)C1)F C12(Sc3scc(C(=O)NC(=O)Cc4cc[nH]c4)n3)CC1CN(N)C2.c1(C=O)ccc(F)cc1 C1(CNC(C2(NC(C)=O)CCCC2)=O)COCCN1C(c1sccc1Br)=O C(=O)(C(C)CCCC(C)=O)N1CCN(CC)CC1.c12ccc(cc1)CN2C c1(C(N2C(C(=O)NCC3CN(C)C(=O)C3)CCC2)=O)cc2cccn2cn1 Cn1nnc(=NC2CC3(CCN(C(=O)CCCCC(N)=O)CC3)C2)[nH]1 C1(CCNC(CCC(=C)C)c2nnnn2-c2ccc(F)cc2)CCC2(CC1)CC2 c1(C2c3nnnn32)ccc(Cl)cn1.c1(C(C)NC2CCC2C(N)=O)cn(C)nn1 C12(CCCSC1)CN2.c1(NCC)cc(C2CC2)nn1C C1(NC(C(C)(C)C)=O)CN(C(c2cc(-c3ccccc3F)on2)=O)CC1O CCCCCCCCC(=O)NCCCCC(C)NC(C1CCC(=O)NC1)=O C1(C(N(C2CCN(C(C3CCC(C)O3)=O)C2)CC2CC2)=O)CCCC2(CCC2)C1 CC1(C)C(CNC(=O)CN2OC(C)(C)CC2=O)CCN1C(C1C2CC3C(C2)C13)=O c1(NC(C2CCCCN2C(=O)CCN2CCCCC2)=O)cc(F)nc(F)c1 c1(CC)cnc(C(=O)NCC2CCC(NC(=O)CN3CCCCC3=O)CC2)nc1 C1(NC(c2cccc(CCO)c2)=O)CN(C(C2CCSC2)=O)CC(F)(F)C1 c1(C(N(CC(C)NC(c2cnn(CCO)c2)=O)CC)=O)ccn(C)c1C N1(C(c2nc(OC)oc2)=O)CC(CO)C2(C1)CN(C(c1cccn1C1CC1)=O)C2 C(CC(CC)C(=O)N1CC2CC(NC(=O)CC3(c4ccon4)CC3)C1C2)=CC C1(NC(C2(OC)CCC2)=O)CCC(N(C)C(c2ccccc2NC)=O)CC1 c1(C(C)C)cc(C(N2CC=CC2CNC(=O)CC(O)CN(C)C)=O)nn1C c1(NC(C2(CNC(C(C=C)C)=O)CCCC2)=O)sc2c(c1C#N)CCCCC2 N1(C(C(CCOC)C)=O)CCN(C(C2CCN(C(=O)CC)C2)=O)CC12CC2 S(=O)(=O)(c1ccc(F)c(Cl)c1)N1CCC(C(F)(F)F)(N(C)CC2CC(C)(C)C23CC3)C1 C1(C(N2CCC(NC(=O)Nc3ccc(O)cc3)CC2)=O)CCCC2(CCC2)C1 CCC(C(=O)NCC(O)CN(C(=O)Cc1ccc(CO)cc1)C)C(C)(F)F c1(NC(C2(C)CCCN(C(c3cocn3)=O)C2)=O)ccc(Br)c2ccccc12 N1(C(c2cnc(C)[nH]2)=O)CC2CCC1CN2C(=O)Cc1csc2sc(C)cc12 c1(OCC(N2CC(CC(C)NCC3COCCO3)C2)=O)cncc(Cl)n1 C(C(C(C)C)NC(=O)C=NOC)(c1ccccc1)NC(c1cnc(CC)s1)=O c1(OCCN(C(=O)C)CC#C)ccc(C)cc1.c1(CS(=O)(=O)CC)cccs1 N1(C(C=CCCC(C)C)=O)CCSCC1C(=O)N(CCC(C)(C)O)C N#CC1CN(C(c2csc(C(=O)N(c3ccc(Br)cc3CO)CCO)n2)=O)CCO1 C1(C(=O)NCCCS(C)=O)CCN(C(C2(C)CCCS2)=O)CC1 C1(C#CC(=O)N2CCCC2CNC(c2cc(C(F)(F)F)on2)=O)(CC)CC1 n1(CC(=O)NCCNC(C2CC3CC3C2)=O)ccc2ccccc2c1=O N12CCCC1C(C)C1CC1C2=O.n1(C)cc(COC2CCC2)nn1.C1(N)CC1(C)Br C(CCCCCCO)NC(c1ccc(-c2cn(Cc3nccs3)nn2)cn1)=O c1(OCC(=O)NCC)ccc(C(N2CC(NC(=O)C(F)OC(F)(F)F)C2)=O)cc1 C1(C2CCOCC2)(NC(COCCC=C)=O)CCN(C(C2CC2C=C)=O)C1 CC1OC2(C(N3CCC(CN(c4ccccc4)CCO)C3)=O)CC1C2 c1(C(N(C)CCN(C)C(C2CCC(C(F)(F)F)CC2)=O)=O)ccc2scnc2c1 CC1=C(C(=O)NC2CC(C(=O)NC3(C)CC3)C2)SCCO1.C1(C(=O)N)CCC(C)C1 N1(CC)CCC(C(=O)NCCCCNC(c2csc(-c3cnn(C)c3)n2)=O)C1 c1(C(=O)NC2C(CNC(C(C(C)(C)C)OC)=O)C2)c(Br)ccc(F)c1N c1(C(N2CC(C)(C(=O)NCC3(F)CCC3)C2)=O)cc(I)cnc1Cl c1(CC(=O)NCCC2CCN(C(C(C)=C3CC3)=O)C2)ccc2cnccc2c1 CC(C)P(=O)(CC(=O)NC1CCC(CNC(c2csc(C(N)=O)n2)=O)C1)C(C)C Cc1cc(C(=O)NC2CC(NC(c3ccccc3)CCO)C2)c(C)[nH]1 C(=O)(C(F)(F)C(F)(F)C(F)F)NC1CN(C(CNC(C=C)=O)=O)CC12CC2 c1(C(C)(C)C)n[nH]cc1S(=O)(=O)NC1CS(=O)(=O)C1(C)C c1(C(N2C(CNC(C3CCSCC3)=O)CCC(C)C2)=O)cnc2[nH]cncc1-2 c1(NC(c2cccc(C)c2)CNC(C(C(=C)C)(C)C)=O)cc2nnc(C)n2cn1 N1(C(C(C)n2ccnc2)=O)CC(CNC(C2CCN(CC3CC3)CC2)=O)C(O)C1 O=C1CC2(CCN(c3cc(N)ncn3)CC2)CN1.C1(CN)CC2CCC1O2 C(=O)(C1=Cc2ccccc2OC1)N1C2CC(NC(=O)C=CC(F)(F)F)CC1CC2 c1(C(=O)NCCC2OCCN(C(CC(CN(C)C)O)=O)C2)cc(F)c(F)cc1N c1(C(=O)NC2CC(O)(CNC(C(CSC)O)=O)C2)cccc2sncc12 C12(NC(CS(C)(=O)=O)=O)COCCC1CN(C(c1cnc3[nH]cnc3c1)=O)C2 n1(COC)nccc1C(=O)NC1CC1CNC(=O)COC1(C)CCCC1 C12(C(=O)NCc3ccc(C(N(C4C(C)CC4)C)=O)o3)CCCC1C2(F)F c1(C(N2CC(C(C)NC(Cc3cc(C)sc3C)=O)C2)=O)cc(C)n(C)c(=O)c1 N1(C(=O)Cc2ccsc2Cl)C2CCC1CC(C(N1CCCC1CF)=O)C2 c1(C(=O)NCC2C(CNC(C3(C(=O)NC)CCC3)=O)C2)coc2ccc(Cl)cc12 N1(C(Cc2ccc(C)o2)=O)CCS(=O)(=O)C(CCNC(=O)C2=CCC(C)CC2)C1 c1(NCCN(C)CCO)ccc(S(=O)(=O)N2CCC(OCCCO)C2)c(Cl)c1 C1(CNC(c2cc3[nH]ccc3s2)=O)CC2CCC1N(C(C1CCCSC1)=O)C2 c1(-c2c(N)csc2)ccc2c(c1)COC21CN(C(C2CCc3n[nH]cc3C2)=O)C1 Cc1cc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)C2CC2)n(C(C)(C)C)n1 C1(O)(CN(C)C(c2conc2C2CC2)=O)CCN(C(=O)C(C)(C)CC2CCC2)C1 c1(N(CC(C)C(C)(C)C)C)cccc(S(=O)(=O)NCc2ccc(Cl)o2)n1 O=C(C#CC1CCC1)N1CCC(CC2CN(C(=O)CC3CCCC4CC34)C2)CC1 C=CC(C)(CCOC)C(=O)NC1CCN(C(=O)NC2(OC)CCCCC2)C(C)C1 N1(C(CCCNC(C)=O)=O)CCCC(C(=O)NCC2CC3CCC23)C1 Cc1cc(C)c(CC(N2CC3(CCN(C(=O)C=Cc4cc[nH]c4)C3)C2)=O)c(O)n1 N1(C(C(C)C)=O)CCCCC1C(=O)N(C)CCN(C(=O)Cc1cccc(F)c1)C C1(CNC(C2C(NC(C3C(CC)C3)=O)CC2)=O)CCCCCCC1 N1(C(C(=O)NCC=C)C2COC2)CCOC(C(F)(F)F)C1C c1(C(N2CC(N(C(CC3(C(=C)F)CCC3)=O)C)C(O)C2)=O)cnc2sccn12 c1(OC)ccc(C=CC(N2CCC(NC(=O)C(C)C(F)(F)F)C2C)=O)c(C)c1 N1(C(CCC(=O)OC)=O)CC(N(C(=O)C(C2CCCCC2)N(C)C)C)C2(CC2)C1 CCCC(C)(O)CC(=O)NC1CCCCN(C(c2ccc(F)nc2)=O)C1 N1(C(c2c(CNC(C3C(C)SCCC3)=O)ocn2)=O)CCCC(C#N)C1 c1(C(=O)NC2(CNC(C(C)(O)C3CCC3)=O)CCOCC2)nc2ccccc2[nH]1 C1(CNC(CCCOCCOCC)=O)CCCN(C(=O)C(c2ccnn2C)O)C1 CC(C)C(O)C(F)(F)C(=O)NC1(C2CCN(C(C3CC4(CC4)CN3C)=O)C2)CC1 C(=O)(C1CCc2ccccc21)NC1CCCN(c2snc(C(C)(C)OC)n2)C1C C1(OCC)CCCC(C(=O)NC(CO)C(C)NC(=O)COCCOCCO)C1 C1(CCNC(C23CC(F)(C2)C3)=O)(OC)CN(C(=O)CCC2CC2(Cl)Cl)C1 N1(CCOCCN(c2cccc([Si](C)(C)C)c2)C)CCCC(C2CCCCC2)C1 Cn1cc(C(=O)NCCC2CCN(C(C3(CO)CCCO3)=O)C2)c(O)nc1=O N1(C(C23OCC(C)(C2)C3)=O)CC2CCC(C1)N2C(C1(C)CC(F)(F)C1)=O C=CC(C)(CCOC)C(=O)NC(Cc1ccco1)C(=O)N(C)Cc1csnc1C C1(C(=O)NCC23OCC(NC(=O)CCc4ncc[nH]4)(C2)C3)COC2COCC12 c1(NC2CCCC(CC(=O)OC)C2)cnc2c(c1)c(Br)nn2C c1(C(=O)NCC(C2CCC2)NC(c2[nH]c(=N)sc2)=O)cc2ccccc2cc1F C1(CNC(=O)CC23CCCC2C3)CC2CN(C(c3csc(F)c3)=O)CC12 CC1(CNC(c2csc(C3CCCO3)n2)=O)CCCN1C(=O)COCCCF c1(CNC(CC2CN(C(C=CCOC)=O)C2)=O)cc2cc(Br)ccc2s1 c1(C(=O)NCCNC(c2nc(C(C)=O)c(C)o2)=O)cc2cnccc2cc1F C1(C(N2CCC(NC(C=CC)=O)C2)=O)CCCCC1C1CC1 S(=O)(=O)(c1ccccc1)N1CC2C(CNC(c3cnnc(Cl)c3)=O)(C2)C1 C=CCCCC(C1CC1)NC(c1cn(CCNC(C2(C)CC(F)(F)C2)=O)cn1)=O c1(C(=O)NC2C(NC(C(CCC)C)=O)C2)c(CC)cccc1F c1(OC)ccc(CO)cc1C(=O)NC1CCC1CNC(=O)C(C1CCOCC1)O N1(C(C=NOC)=O)CCC(C)(CNC(c2ccc(C#N)s2)=O)C1 Cc1cc2ccc(C(=O)NCC3(NC(=O)CC=CC(C)(C)C)CC3)cn2c1 c1(C(N(CCCC)CCNC(c2ccco2)=O)C)nc(CC)no1 N1(C(C2CC(C)(CC)C2)=O)CCC(NC(c2csc3nccn23)=O)C12CC2 N1(C(c2nc(C)sc2)=O)C2CCC1CC(CNC(c1ccnnc1Cl)=O)C2 N1(C(C=COCC)=O)CCC2(CCCC2NC(c2cc(C3CC3)ncn2)=O)C1 C1(C(C2CC2)NC(c2cccc(OC)c2)=O)CCC(n2cc(C3CC3)nn2)CC1 C=C(C)C1CCC(C)=CC1CC(N1CCC(C)(NC(=O)CC2CC(C)C2)CC1)=O C1(CC(=O)NCC2CN(C(c3cnc(C)o3)=O)CC2(C)C)CCn2cncc2C1 C1(SC)CN(C(=O)CC2CCCCC2O)CC1NC(C1(C(F)F)CCCO1)=O C(c1ccc(F)cc1)=CC(=O)NC1(CCNC(COC)=O)CC1 CC(c1ccccc1)=CC(=O)N(CCC(C(C)(C)C)NC(C1(CF)COC1)=O)C C1(CC(N)=O)CN(C(=O)CC2CCN(C3CC3)CC2)CCC1NCc1ccsc1 Cc1nc(C2CC2)[nH]c1C(=O)NCCC(O)CNC(=O)C(c1cccc(F)c1)C C1(NC(=O)CC2CCCOC2)CCSC12CN(C(c1ncc3[nH]ncc3n1)=O)C2 Cc1cn2c(n1)CC(C(N1CC(C(C)NC(c3cc(Cl)sc3Cl)=O)C1)=O)CC2 Cc1ncc(C(N2CCN(C(=O)C(N)Cc3ccc(O)c(F)c3)CC2)=O)c(O)n1 C1(C(N(CC(C)(C)NC(=O)C(F)=C(C)C)C)=O)CC(C(F)(F)F)CO1 N1(C(C2C3CN(Cc4c(C)n[nH]c4)C2C3)=O)CCn2cccc2C1 c1(CC(N2CCC3CC23C(=O)NC2CC(O)(CO)C2)=O)ccc(F)c(F)c1 C(=O)(C(C(C)O)N)NC(=O)C(C)(C)C.C12(C(=O)NC(C)CNC)CC(C1)C2 C1(NC(C)=O)C2CCN(C(=O)C(c3ccccc3)n3cccn3)CCC12 Cc1coc(C(C)C)c1C(N1CC(NC(C23CCC2C3)=O)C(F)C1)=O c1(C(=O)NCCN(CCC)C(C2(Cl)CC23CCC3)=O)c(Cl)ccc(F)c1F Cc1nncn1CCCNC(=O)CC1(F)CN(C(=O)C(O)CN(C)C)C1 C(C)(C)(CC(C(=O)NCCc1ccc(F)cc1)OC)N(CCCF)CC c1(C(C)=O)ccc(C(=O)NC2CCCCC2CNC(=O)CCNC(=O)CO)nn1 N1(S(c2cccc(C#N)c2)(=O)=O)CCc2nc(C3=CCC(O)CC3)sc2C1 C1(C(C)C)C(=O)O1.C1(NC(CCOCCCNC(C)=O)=O)CCC(C(N)=O)CC1 c1(C(=O)NC2(CO)CN(C(c3cc(Cl)on3)=O)C2)ncn2cccnc12 Cc1c(C(=O)NC2CCN(C(C3CC=CC3)=O)C(C)C2)nn2cccnc12 c1(N2CCC(CNC(C3(CC(C)C)CCCC3)=O)CC2)c(F)cccc1[N+](=O)[O-] C(=O)(C(=O)CC(C)CC)N(C(C(=O)NC(CCCC)C(=O)N(C)C)C)C c12ccc(nc1)[nH]2.n1(C(C)(C)C)cc(CNC2CCCC2)cn1 N1(C(c2cc(CC)sn2)=O)CCOCC(NC(=O)C=CC2CCCC2)C1 C1(C(=O)NC2(C(=O)OC)CC2C)CCCN(C(C2NC(=O)OC2C)=O)CC1 O=C1CS(=O)(=O)CC(C(N2CC(O)(CNC(c3ccnc4ncnn34)=O)C2)=O)N1 c1(C(=O)NC)ccc(C(=O)NCCCN2CCC(C(=O)OC)C2)cc1F c1(NC(C(=O)Nc2cc(Cl)ccn2)=O)ccc(Br)c(Cl)c1 CCCC(O)CC(=O)N1CCN(CCCNC(C2CC23CCOCC3)=O)CC1 N1(C(CC(C)OC)=O)CCCC(C)(CNC(C2CS(=O)(=O)C2)=O)C1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N(C1CC2CCC1N2)C(c1c(C)noc1)=O C1(NC(C(CCC)(C)O)=O)CN(c2ncc(O)cn2)CC2(CCC2)C1 C(=O)(C(CNC(=O)C(C)S(N)(=O)=O)(CC)CC)N1CCN(C(C#C)C)CC1 C(c1cccc(Cl)n1)=CCO.C1(CCN(C)C)CN(C=O)CCO1 C#CC1(C=C)COCCN1Cc1n[nH]cc1Br c1(OC)ccc(F)c(CC2CN(C(c3ccccc3Cl)=O)CC(C(=O)O)C2)c1F C1(NC(=O)CCc2ncccn2)C2CN(C(=O)CCc3nc[nH]n3)CC12 N1(C(C=C(CCC)C)=O)CCCC(C)C1CNC(C1(C)CCC(F)(F)C1)=O Cc1ccc(OCCC(N2CCC(Nc3ccc(N)cc3)C(C)C2)=O)c(C)c1 c1(-c2ccc(C#N)nc2)cccc2c1CCN(S(=O)(=O)CCn1cncn1)C2 C1(NC(C(C)(C)NC(=O)NCCC)=O)CN(C(c2cccc(=O)o2)=O)CC1C CCC(O)C(C)C(=O)NCC1CN(C(c2cn(C)nc2C)=O)CC1N(C)C C12CCCN(C1)C2=O.c1(CCC)nnc(N(c2nc[nH]n2)CC)s1 C1(C(C(=O)NCC(C)N(C)C(C2(C(F)(F)F)CC(O)C2)=O)OC)CCCCCC1 c1(C(N(CC(CNC(C(CC)CCOC)=O)O)C)=O)cc2c(nc1O)CCSC2 C1(C(C)C)CN(C(C2(CO)CC2(F)F)=O)CCN1C(=O)C(C1CCCCCC1)C Cc1c(C(N2CC3CCC3(NC(=O)CCC(C)(F)F)C2)=O)cccc1N c1(NC(C2CC(NC(c3ccc(OC)s3)=O)C2)=O)ccc(F)c(C(F)F)c1 CN1CCC(F)(CNCCOCCn2cc(C(=O)NC3CC34CCCC4)nn2)C1 C12(OC)CCC(C(N3CC(NC(C4(F)CCOC4)=O)C4CCCC34)=O)(CC1)CC2 C(CN(C)C)(C(=O)NCCC(F)F)NC(CN(C(C)C)C)=O N1(C(CCC(C)C)=O)CCCN(C(C2CC3(C)CC2CO3)=O)CC1CO C1(CC)CCN(C(c2csc(C#N)c2)=O)C1C(=O)Nc1cccc(OC)c1 C12CCN(C(c3nc(CC)n(-c4cccnc4F)n3)=O)C3CCC(CC13)C2 c1(C(N(CCC(CC)(C(=O)OC)CC)C)C(=O)NC(C)C)cccc2c1CCCC2 C1(n2cc(C3(C(=O)NC)CCC3)nn2)CCCCC1NC(C1CC1(Cl)C(=O)OC)=O N1(C(CC2(OC)CCCC2)=O)CCCC(N(C(=O)CC(C)c2ccccc2)C)C1 N1(C(c2ccc(F)cc2Cl)=O)CCC2(CCCCN(C(C34CSCC3C4)=O)C2)C1 c1(C(N2CCC(NC(C3(CCOC)CC3)=O)C2)=O)cc(Br)cc2c1OCO2 C1(C(N2CCN(C)CC2CNC(=O)CC(F)(F)Cl)=O)CCc2[nH]nc(O)c2C1 C=C(C)CC(C)C(=O)N1CCCCC1C1CCN(C(=O)CCCOCCC)CC1 CC1=C(C(=O)N2CC3CC2C3NC(c2ccc3ccoc3c2)=O)C(=O)OC1(C)C C(=O)(C(C)(C)C(=O)N1CCN(C)C(CNC(c2nc(=O)n(C)[nH]2)=O)C1)N(C)C CCC(CC(=O)NC1CCN(C(=O)C=C(C)c2cccc(Cl)c2)CC1)C(C)(C)C C1(F)(C(N2CCC(O)(CCNC(CN(CC(C)(C)C)C)=O)C2)=O)CC2(CCC2)C1 N#Cc1ccnc(C(N2CC3C(CNC(=O)C=CCF)C3C2)=O)c1 Cc1nc(C(=O)NCCC2CCC(NC(=O)C(C)(Cl)Cl)C2)sc1C N1(C(c2onc(C)n2)C)CCCC(C2CCCN(C(c3cc(C)nn3C)=O)C2)C1 C1(NC(C2CC(C)(NC(c3c(CC)ocn3)=O)C2)=O)CCCCC1C(N)=O C(=O)(CC1CC(O)c2ccccc21)N1CCCCC(CNC(CCCSC)=O)C1 N1(C(C(C2CCC2)OCC)=O)CCCC1(C)C(N1CCCC(CN=[N+]=[N-])C1)=O NS(=O)(=O)c1cccc(C(=O)NCCC2CCCN(Cc3cnc(Br)s3)C2)c1 Cc1nn(C)c(NC(C2(CN)CC2)=O)c1Br.c1(CN)sccc1C(=O)N(C)N(C)C n1(CC(=O)NCc2occ(C(=O)NCCCC3CC(C)C3)c2)ncn(C)c1=O C(=O)(C(CP(C)(C)=O)C(F)(F)F)N(C)CCC1CC1.C(C)(C)(C)OC=O N1(C(c2cncc(OC)c2)=O)CCCC(NC(=O)C=CC2CCCCCC2)C1C CCC(CNC(C1Cc2nccn2C1)=O)(CC)C(=O)N(C1CC(C(C)C)C1)C Cc1cccc(CN2CCC(O)C2C(=O)Nc2ccc(Cl)c(F)c2)c1O N1(C(Cn2cnc(=N)[nH]2)=O)CC(NC(=O)C2=C(Cl)CCCC2)C(N=[N+]=[N-])C1 N1(C(C=C)=O)CCOC2(CCN(Cc3cc(OCC(F)(F)F)ccc3F)CC2)C1 c1(C(=O)NCC(C(C)C)NC(C2(C)C(C)(C)C2)=O)cc(Br)c([N+](=O)[O-])[nH]1 c1(N2CCC(C3N(C(c4ccsn4)=O)CCCC3)C2)cc(C(F)(F)F)nc(Cl)n1 N1(CC(N2CCOCC2)C)CCn2cc(C(N3CC4(CCC4)C3)=O)nc2C1 N1(C(CN(C2CCC2)C)=O)CCC(CCCCNC(C2CCCCO2)=O)CC1 N1(C(C2(CO)CC(C)(C)C2)=O)CC2CC(C(=O)NC(CO)CCC3CC3)(C2)C1 C1(NC(C=CC2(C)CCOCC2)=O)CN(C(=O)CC2(O)CCCC2)CC1C1CC1 c1(C(=O)NC2C(NC(C(CNC(C)=O)C(C)C)=O)COC2)cc2ccncc2[nH]1 C1(N(C(c2cc(F)ccc2OC)=O)CC)CCCN(C(=O)OC(C)(C)C)C1C Cc1ncc(NCc2nn(C)c(C)c2C(=O)O)c(C#N)n1 c1(C(CO)NC(C2C=CC(NCc3ccnc(Br)c3F)C2)=O)ccc(F)cc1F C#CC1COCCC1N1CC2C(C(=O)N(c3ccccc3Cl)CCCO)C2C1 C(C)(C)(CCCNC(C1(C#N)CC1C(F)(F)F)=O)NC(C1C(CC)C1)=O C1(CC(=O)NCc2nc(C)oc2)C2CCCC2N1C(c1sccc1C#N)=O c1(C(N2CC3C(NC(C=CCCC(C)C)=O)(C3)C2)=O)ccn2[nH]c(=N)nc2c1 C(C(CC(F)(F)F)NC(C12CCC(C1)C2)=O)NC(CC1(CC)CCC1)=O N1(C(CCCCSC)=O)CCC(N(C)C(c2ccnc(CO)c2)=O)C(C)C1 c1(OCCOC)ncccc1C(=O)N(C)CC1CCN(C(=O)C(F)C2CCC2)C1 c1(CC(N)=O)ccc(C(=O)N(C2CCN(C(C3(F)CCCCC3)=O)C2)C2CC2)cc1 c1(C(=O)NC23CC(NC(=O)C=Cc4cnc[nH]4)(C2)C3)ccc2snnc2c1 c1(NC(C)=O)ccc(C(=O)NC23CC(NCc4c[nH]cc(Br)c4=O)(C2)C3)c(Cl)c1 CC1=CCC(C(N2CCC(C)(NC(=O)CCc3cc(C)[nH]n3)C2)=O)CC1 C12(CNC(C3N(Cc4cnc(C(=O)OC)nc4)CC=C3)=O)CCCN1CCC2 C(CCC(C(=O)NCC(F)Cl)NC(c1nonc1N)=O)OC Cc1[nH]nc(-c2nc(-c3cnc(CC4(C)CCCO4)o3)no2)c1C Cc1cc(N(c2ccccc2)CC(=O)NC2CCCOC2CC(C)C)c(F)cc1Cl N1(C(CC2(O)CC(C)(C)OC2)=O)CCC2(CC1)OCCC2NC(=O)C=CI c1(C(=O)NCC(CCOC)NC(C2OCC2(C)C)=O)ccc(C(=O)OC)cc1F CN1CCC(C(=O)NCC#CC(=O)NC2CCCC2C(N)=O)C1 c1(CNC2C3CN(C(C(CC)N(C)C)=O)CC32)ccccc1[N+](=O)[O-] c1(N(CC(CN(C(c2c(OC)cccc2)=O)C)O)C)nccc2scc(Br)c12 c1(C(=O)NC2CCC(NC(Cc3c(C)cco3)=O)C2)cc2c(nc1O)CCCC2 C1(Cl)(C(=O)OCc2cc(C#N)oc2)C2CCC(=O)C12 C1(NC(c2c(C)cc(C)o2)=O)CCN(C(=O)CCCCN(C)C)C(C)C1 Cc1cc(Cl)ccc1OCC(=O)N(C1CCN(C(c2ncnn2C)=O)C1)CCO C(C(=O)NC(=O)C(F)F)(C(F)(F)F)Nc1ccc(C(=O)OC)cc1 C1(CNC(CCC(C)SC)=O)CCCCCN1C(=O)CN1CCN(C(C)C)CC1 N1(C(C2(C#C)CC2)=O)Cc2nccn2CC(NC(c2cnc(C(C)(C)C)s2)=O)C1 C1(N(C(C(C)N2CCCC2)=O)C)CCCN(C(c2cnc(C(F)F)s2)=O)C1 N1(C(C(=O)NCC)=O)CCCCC(CNC(c2cnn3ccn(C)c23)=O)CC1 c1(C(=O)NC2CN(C(C3CCCS3)=O)CC2O)cc(Br)cc2cccnc12 C1(NC(CSC(C)(C)C)=O)CN(C(c2cncn2C2CC2)=O)CC12CC2 C1(C(=O)NCC2CCC(NC(c3ccncn3)=O)C2)CC2(CCC2)C1 c1(C(N2CCC(Oc3cc(F)cc(F)c3)CC2)=O)cc(F)cc(I)c1 c1(C(=O)NCC2(O)CCCN(C(C(CC)C3CC3)=O)C2)cc2ccccn2n1 CC1CCN(C(=O)C(C)(C)C(=O)N(C)C)CC1CNC(=O)C(C)(C)F CCCCCS(=O)(=O)CC(=O)N(C)CC1CCN(C(=O)C(C2CCCCC2)F)C1 c1(C(N(C(CCNC(C(CCCCC)O)=O)C)C)=O)cnc2ccnn2c1O C(=O)(CC(C)(C)C)NC(C)C(=O)NCC#CCN(C(=O)CCc1cc[nH]n1)CCC N1(C(C(F)=C(C)C)=O)CC(C(=O)NCc2ccc(C#N)cn2)C(C)(C)C1 CC1CCCC(C(=O)NC(C)C(=O)NC2(c3nn[nH]n3)CC2)C1 C(=O)(C1CCc2snnc21)NC1CCC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 CCCCC(C(=O)N1CCC(CCO)C1)NC(=O)C(C)n1ccnn1 Cc1c(Br)ccc(NC(C2(O)CCN(C(c3c(F)cc(Br)cc3Br)=O)C2)=O)c1F C(N=C(NC(C)C)N1CCC(O)C(C)C1)c1c(C)cc(C)cc1C C1(C2CC2)(CN2C(CO)COCC2)CN(CC2CC3C=CC2CC3)C1 c1(NC2CCCN(CCn3ccc(CC(=O)OC)n3)C2)nc(C)cc(C)n1 c1(CNC(c2cc(F)ncc2NC)=O)cc(C)cc(NC2(COCC)CCC2)n1 C(=O)(C(C)CC(C)(F)F)NC1(C)CCN(C(c2cccc(NC(C)=O)n2)=O)C1 C12(NC(C=CC=CC)=O)CCCCC1CN(C(C1CC3(CCC3)CO1)=O)C2 O=C1CCN(Cc2nc(C(F)(F)F)co2)C(=O)N1CC12CCCC(CO1)C2 N1(C(C(n2cc(Br)cn2)C)=O)CC2CC1C2NC(=O)Cc1ccns1 Cc1ccc(CNC(C2CC2C(=O)O)=O)nc1.c1(C(c2ccccc2)N)ccccc1 c1(OC)ccc2c(c1)C(C(=O)N1CC3CCC(C1)N3C(c1csc(S)n1)=O)CC2 c1(N)cc(F)ccc1-n1cccn1.C12CCCN(C1)C2.C1(C(=O)OC)CC(N(C)C)C1 Nc1cccc(C(=O)NCC2(O)CC(CNC(=O)C(C3CCCCCC3)O)C2)n1 c1(C(N2C(CN(C(c3cc(C(N)=O)c[nH]3)=O)CC)CCC2)=O)cc2n(n1)CCO2 C1(C(N2C(C)(CCC)CC2)=O)CN(C(=O)C=Cc2ccncn2)CCC1(C)C c1(C(N(CCCCNC(=O)CCN2C(=O)CCC2=O)C)=O)cccc(Cl)c1F C1(NC(C2(CNC(C3CC4C=CC3CC4)=O)CC23CCC3)=O)CC2CCC1CC2 C1(C(=O)NC(c2nn[nH]n2)C2CCOC2)CCCSC1 c1(C(N2CCN(c3nc(SC)nc(C)c3)C(C)C2)=O)ccc(F)c(Br)c1F N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CC2CC1CN(C(=O)CCC(N)=O)C2 CCN=c1ccc(C(N2CC(O)(CNC(=O)CCn3cccn3)C2)=O)c[nH]1 C=C(C)C1OCCC1C(N1CC2CC1C2C(=O)NC(c1cn[nH]c1)C)=O C(CC#CC(C)(C)C)NC(C1(C#C)CN(C(C2CC2C(F)F)=O)C1)=O c1(C(=O)NCCC2(CNC(CC(C)n3cccn3)=O)CC2)cc2ccncc2s1 C(=O)(CC1=CCCC1)NCC(C)C(=O)NCC1(C(N)=O)CC1 CC(C)(CCC(=O)NC1CCCCN(c2ncns2)C1)[N+](=O)[O-] c1(CC)cc(OC)ccc1C(=O)NCC1CCN1C(=O)C(C)(C)c1cncs1 CC1CC(c2cccnc2)N(C(=O)COc2cccc(Cl)c2)CC1C N1(C(CCC)=O)CC(NC(C2(C)CC(C)(C)C2)=O)CC(COC)C1 N1(C(CC(=O)N(C)C)=O)CC2(CNC(c3cc(Cl)cc(F)c3F)=O)CCC1CC2 N1(C(c2cc(OCC)n[nH]2)=O)CCC(N(C(C2CC2(C)Br)=O)CC)CC1 N1(C(C(c2c(C)noc2Cl)CC)=O)CCOC(CNC(=O)CSCCC(C)C)C1 C1(C(=O)NCC2(CNC(=O)Cn3cnnc3O)CCC2)C2CC3C(C2)C13 N1(C(C2C(C)N(C(C3CC4CCC3CC4)=O)CCC2)=O)CC(C2CCCC2)C1 C1(CC=C)(C(=O)NC(CCOC)C(C)C)CCCN1C(=O)CC1CCCC12CC2 c1(Nc2c(OCC)cccc2)c(C(=O)OC(C)(C)C)cnc2c1cnn2C c1(NCC(C)(C)CSc2ccccc2)ncnc2c1cnn2-c1cccc(F)c1 C(CCC(C)C)(C(=O)NCCC(C(C)C)NC(=O)CCC(=O)N(C)C)NC(=O)OC C1(C(N(CCCNC(CN2C(C)CCC2)=O)C)=O)CC2CCCCCC12 CC(C)CC(C)C(=O)NCCCN(C)C(C12CCC(C(F)F)(CC1)C2)=O C1(O)(CC(=O)Nc2cncc(Br)c2)CCN(Cc2cnc(Cl)s2)C1 c12ncc(cn1)NC2c1nnnn1C.c1(CC)cccnc1C(C)(C)C CCCC(C(=O)N(CCCNC(c1ccnc(C)n1)=O)C)OC.c1(SC)ccccc1 O=C(C1SCCc2ccccc21)NCC12CC1CN(CCC=Cc1ccccc1)C2 CCCC(C)CC(=O)NCC(CC1CC1)C(=O)NCC(C1CC1)SC c1(CC)nc(C)c(C(=O)NCC2CCCN2C(c2cccc(SC3CC3)c2)=O)s1 C1(NC(CC(=O)OC)=O)CCCN(C(=O)Cc2cccc(OC3CCOC3)c2)C1 C1(CC)CN(C(=O)CN(c2csnn2)C)CCN1C(=O)CCCCC1CC1 C(CCCC(F)(F)F)NC(c1c(CNC(CCc2ncn(C)c2)=O)cco1)=O CC1=C(C)CC(C(=O)N(CCCNC(c2cc(C)sc2C)=O)C(C)C)CC1 C1(CC(N2CC=CC(NC(Cn3c(CC)ncc3)=O)C2)=O)Cc2ccccc2O1 CC(CN(c1cccc(Cl)c1)C)CCC(=O)N(C)CCNC(=O)CCS(C)(=O)=O c1(C(=O)NC2C(NC(c3c(C)ccc(Cl)c3)=O)CCC2)cc(Cl)c(F)c(Cl)c1 C1(CNC(c2n(CC)nnc2)=O)CC(O)CN1C(c1ocnc1C1CC1)=O c1(CC(=O)OC(C2CCC(Oc3ccncc3)C2)C)cc(Cl)sc1Cl c1(C(N2CCC(c3cn(CCOCCO)nn3)CC2)=O)cc(F)c(Br)cc1[N+](=O)[O-] c1(C(N2CC(OC)(CNC(c3n[nH]cc3Cl)=O)C2)=O)ccc(-n2ccnc2)cn1 C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)COC)CCS(=O)(=O)CC1 Cc1cnn2c1CN(C(=O)NCCC1CCCCC1(F)F)CC2 C(=O)(C1COCc2ccccc21)NC1CCN(C(c2c(SC)nc(O)nc2C)=O)C1 C(N=c1[nH]c(=NC(C)C2CSC2)[nH]c2cc[nH]c12)c1cc(OC)c([N+](=O)[O-])cc1 c1(C(=O)OC)cccnc1NCCCC1CCCN1C(=O)Cc1ccc(Cl)cc1 N1(C(C(CC(=C)Cl)NC(CC=CC=C)=O)=O)CCC2CCCCC12 c1(CC)cc(Cl)ccc1C(=O)NC1COCCC1NC(C1CCC(=O)N1C)=O c1(C(=O)NCC(CC)NC(=O)CCS(C)=O)nn(C)cc1Cl C1(C(N(C(C#C)C)C)=O)CC2(CC2)C12CCC2 CCCCCC(C)CC(=O)NC1CCN(C(=O)CC2CN(C(C)=O)C2)CC(O)C1 N1(C(C2(C(=O)NC)CC2)=O)C2CCC1CN(C(=O)C(c1ccc(Cl)cc1)=O)C2 C1(C(=O)NC2CC(OCC)C2)N(C(C2CCCCC(=O)N2)=O)CCCC1(C)C C(=O)(C1=C(C)OCCC1)N1C(C(=O)NC(CC=C)C2CC2)C2CCC1C2 c1(C(=O)NCC(C)CN(C)C(C2CS(=O)(=O)CCO2)=O)cnn2cccnc12 C1(CNC(c2cc(Cl)c[nH]2)=O)COC(CNC(C2(n3cccn3)CCC2)=O)C1 c1(CC(=O)NCCN(C(CC(=C=C)C)=O)C2CC2)ccc(F)cc1C N1(C(CCC(C)NC(C23CCCC2C3)=O)=O)CC2(COC(=O)N2C)C1 c1(C(=O)NCC(C2CCC2)NC(C2CC(C(C)C)C2)=O)cc(C(F)(F)F)n[nH]1 C1(C(=O)NCC(CO)OC)CC(C)CN1C(c1[nH]nnc1C)=O c1(C(=O)NCCNC(C(CCC)O)=O)cnc(C)c(Cl)c1Br C1(CNC(C(C)(C)OC)=O)CCN(C(c2cc3ccccc3[nH]2)=O)C12CCC2 c1(C(N2CCCC(CCNC(CC3(C)CCOC3)=O)C2)=O)ccc(P(C)(C)=O)o1 C1(OC(C(N2CC(C)(OC)C2)CSCCNC(C)=O)=O)CC(C2CC2)C1.OCC N1(C(C(C(C)CC)N(C(C(C2CCC2)OCC)=O)C)=O)CCC(C2(C)CC2)C1 c1(CN2CC(NC(C3CCCC(C)C3)=O)(CO)C2)cc(Br)c(F)cc1Cl N1(C(CC(C)O)=O)CCCCC1C(C)NC(=O)Cc1cccc(F)c1 Cc1cc(C(=O)NC2CCC(NC(C3(C#N)CCC3)=O)CC2)cc(C)c1Cl c1(CNC(C(C)=C(C)C)=O)cccc(C(=O)NCCn2cccnc2=O)n1 N1(C(CN(C)C)=O)CC(F)CC1CNC(C1CC1c1ccco1)=O C(=O)(C1=C(CC)OCCC1)N1CC(NC(c2c(Cl)ccc(C#C)c2)=O)C(C)C1 CN1C(=O)CC(C(=O)Nc2nnc(C(F)(F)F)n(C)c2=O)NC1=O c1(C(=O)NCCN(CC(C)O)C(c2cnc(C(C)C)[nH]2)=O)cnc(Cl)c(F)c1N c1(C(N)=O)cccc(C(=O)NC(C)(CC(=O)O)c2cccc(Cl)c2)c1F C=C1C(C(=O)OC)C1C(=O)N(CCC(=O)OC(C)(C)C)C c1(C(=O)NCC(O)CC(=O)O)ccnn1C(F)F.C1(C(=O)N)(S)CCC1 N1(C(CC(CC)O)=O)CCC2CC1CN(C(c1ccc3[nH]ccc3c1)=O)C2 N1(C(c2c(CC#N)ccs2)=O)CCC2(C1)CN(C(C1CC(C3CCCC3)C1)=O)C2 c1(-c2c(OC)cccc2F)ccc2[nH]c(C(=O)NCC3(C)CC3)nc2c1 N1(C(C(CC=C)C)=O)C2CC1CN(C(=O)Cc1ccccc1CC(N)=O)C2 CC(C(=O)NOCCOCCF)C(C(C)(C)C)NC(=O)OC(C)(C)C c1(OC)ccc(N(C(=O)Cc2ccc(F)cc2)C)cc1 C12CN(CC13CCC3)N1CCOCC(C1)CNC2=O.N1(CC=O)CCSCC1 N1(C(C2C(C)C2)=O)CC(C2CCCN(C(C3C4CCCOC34)=O)C2)C1 CC(C(=O)NC1CC1c1cncs1)(C1CCC1)NC(=O)CCc1ccccn1 N1(C(=O)OC)CCCCC1C1CCCN1CC(=O)C(F)(F)Br C1(N(C)C(C2(CO)CCCC2)=O)CCCCC1NC(=O)C(c1ccccc1)F C(=O)(CCCN1CC(NC(=O)CSCCC(C)C)C1)NC1C(CCC)C1 Cc1cc(F)c(N)cc1C(=O)NCCC(O)CNC(=O)C1=CCCOC1 C1(C)(C(=O)NC2C(NC(c3c(CC)ncs3)=O)CC2)CCCCNC1=O c1(C(=O)NC2CC(F)(CNC(=O)CCC3CCCC3)C2)ncccc1C(F)(F)F CN1CCN(C(c2cc(N)cc(O)n2)=O)C(CNC(=O)CC2CCC(F)(F)C2)C1 C(CCC(C)(C)C(=O)N1CC(C)(C)C1C(=O)OC)NC(C(CC=C)OC)=O C1(CCNC(c2cncc(C)n2)=O)CN(C2CCCNC2=O)CCS1(=O)=O C#Cc1cccc(C(N2CC3C(C(=O)NCc4cc(C)ccc4O)C3C2)=O)c1 CCCCC(CC(=O)N1CCCCC1C1CCC1)NC(c1ccc(C#N)[nH]1)=O c1(CCC(=O)NC23CN(C(C4CC=C(C)CC4)=O)C(C2)C3)cc(F)ccc1F C1(C(N(C(c2cccnc2)C)C)=O)CN(C(c2ccsc2)=O)CC1(F)F c1(C(C)OCC)nc(-c2nnn(CCOC(C)=O)c2C)n(-c2ccnnc2)n1 C1(NC(N2CCC(C)C(C)(O)C2)=O)CC2CCCCC2N1C(=O)C(F)(F)F CC1(C)CCC(C(=O)NCC(C2CCCC2)NC(=O)C(C)(C)c2cc[nH]n2)C1 C1(NC(C2C(NC(c3cc[nH]n3)=O)CC=CC2)=O)CCCN2CCCC12 Cn1cc(C(N2CCC(NC(=O)CC3CCSC3)C(F)C2)=O)ccc1=O N1(CC(N2CCC(O)(CNC(C(C)C3(O)CCC3)=O)C2)=O)CCP(C)(=O)CC1 c1(C(C(=O)NCC2C(CNC(CCC#N)=O)C2)O)ccccc1Br C1(CC)(NCC(F)CN(N2C(C=O)C2)C(c2cnoc2C)=O)CCCCC1 S(=O)(=O)(c1cc(C(=O)N(CC(C)C(C)(C)C)C)co1)NC C1(C#N)(C(N2C(NCc3c(C(=O)NC)scn3)CC2)=O)CCCC1 C(CC(CC)C(=O)NCC(C)CC(=O)NCCC[Si](C)(C)C)=CC N1(C(CCCOC)=O)CCN(C2CN(C(C3CN(C(C)=O)C3)=O)CC2C)CC1 c1(C(=O)NC2CN(C(C3N(CCCC)CCOC3)=O)C2)cc(O)ncc1Br Cc1ncc(Cl)cc1C(=O)NC1CCN(C(=O)Cn2nccn2)CC1C c1(OC(C(=O)N(CC(CC)NC(c2cc(F)c[nH]2)=O)CC)C)ccccc1F c1(C(=O)NC2CCCCC2NC(C2C3COCC23)=O)cnc2ccccn2c1=O c1(C(N(CCOC)CCNC(C2(CCSC)CCC2)=O)=O)c(C)nc(O)nc1C c1(C(=O)NC2CC(O)CN(C(=O)Cc3sc(O)nc3O)C2)cc2cnccc2[nH]1 CCC(CO)C(=O)NC1CN(C(c2cnc(-c3ccc(Cl)cc3)s2)=O)CC1C N1(C(C(C)(C)c2cccnc2)=O)CCOCC(CNC(=O)Cn2ncnn2)C1 C1(OC)CCCC(C(=O)NCCC2(NC(c3cnccc3Cl)=O)CCC2)C1 C1(C)(CNC(c2c(CC)c[nH]n2)=O)CN(C(=O)CCCN(C)C)C(C)(C)C1 c1(C(=O)NC2(C)CCN(C(=O)C=C3CCCCC3)CC2)ccc2ncccc2n1 C(=O)(CCCC(C)=O)NCC(CCOC)NC(c1cccc(F)c1C(F)(F)F)=O CC1(C)OCC2(CCN2C(c2cn(C)nn2)C(=O)NCc2ccccc2)C1 C12(C(N(C3CC(=C)C3)C)=O)CCN(C(C3CC(C)C3)=O)CCC1C2 C1(NC(c2c(C)ncs2)=O)COCCN(C(C2(C#N)CC3CC3C2)=O)C1 C1(NC(C=CC(=O)N(C)C)=O)CCC2CC1CN2C.c1(CC(=O)N)ccsc1.CC=O C(=O)(C1CCc2c[nH]nc21)NC1C=CCC(C(N(C2CCCCC2)CC)=O)C1 N1(C(c2nc(C)c(C)s2)c2nnn(C)n2)CCC12CCCC(C)(C)C2 c1(N(CCC)C)nc(C(=O)NC(=O)CN2CCC(C)(O)C2)cc2ccccc12 c1(C(=O)N=c2[nH]onc2-c2ccco2)cc2ccncc2s1 c1(CC)ccc(C)c(C(=O)NCC(C)(C2CC2)NC(C2CCCC(OC)C2)=O)c1 c1(C(=O)NCCCC(C)NC(c2c(CC)onc2C)=O)cccc(O)c1F C(=O)(CCC(=O)N1CC(C(=O)NCCOc2ccncc2)CC1C)NCC c1(OC(C(C)C)=O)nnc(CSc2ccco2)n1CC1CCS1(=O)=O N1(C(C=Cc2n(CC)ncc2)=O)CC(NC(=O)C(=O)N(C)C)CC12CCOCC2 N1(C(CCC(=C)Cl)=O)CCC2(CCCN(C(=O)CCSc3nccn3C)C2)C1 C(C)(C)(CCC(=O)NCCc1noc(C)n1)NC(Cn1nnc(C)n1)=O N1(C(c2c(C(C)=O)ccs2)=O)CCC(NC(=O)C(C)Cn2ccc(C)n2)C12CC2 C1(C(=O)O)CCC(NC(C2NC3CC2CC3O)=O)CC1 Cc1nc2cc(C(=O)NCCC3CC(NC(=O)CCc4cnc[nH]4)C3)ccc2s1 N#Cc1ccc(N2CCC(NCc3ncoc3C3CCOCC3)C2)c(F)c1 c1(C(N2CC=CC(NC(C(C=C)(C)CC)=O)C2)=O)c(Cl)ccc(Cl)c1O N1(C(C(=O)NCC)=O)CC(NC(C2CCC(F)CC2)=O)C(C)C1 C1(NC(c2ccc3cccnn23)=O)COC2CN(C(=O)C(O)O)CC12 CN1CCC(C)(C(N2CCC(O)C(NC(=O)COc3cccnc3)C2)=O)CC1 c1(-c2n(CCOC)nc(-c3cccc(OC)c3)n2)ccc(Br)c(Cl)c1 C(C1=CCN(C(=O)CC2CC23CC3)CC1)NC(=O)Cc1cc(Cl)sc1Cl c1(C(N2CCCC2CSC)C(=O)NCCOCC)nn(C)cc1Cl Cc1cc(C(=O)NCC2CC(C)N(C(c3ccco3)=O)C2)cc(C)c1 Cc1cc(NC(C)C(=O)NCC(F)(F)CCC(=O)O)c(Cl)cc1C1CC1 C(C(C)(C)C(=O)NCCC1CCC(C)(C)O1)N(C(=O)CCC1CCCOC1)C N1(C(C)=O)CCCCCC1C=O.C1(NC)CC(=O)N(c2ccc(C)cc2)C12CCC2 C(CC(C(=O)N=c1ccn(CC2CC2)[nH]1)NC(N)=O)N1CC(C)OCC1C C12(NC(CCC)=O)CC(C)(C1)OC21CN(C(C2CNC(=O)N2)=O)C1 C1(CC#C)(C(=O)N(CC)CC23CCN(CC2)C3)CCN(C(=O)C(C)SCCCC)C1 c1(C(=O)NCCC2CCC(NC(CC3(C)CC3)=O)C2)ccc(Cl)cc1 C1(CC)CCCCC1OCC(N1CCC(N(C(=O)C=Cc2sccc2C)C)C1)=O Cc1cc(Br)cc(C(N2CCCCC(C)(C)C2)=O)c1C c1(CNC(=O)Nc2nc(C)c(C(C)C)s2)ccc2c(ccn2C)c1 CC1=NOC(C(=O)N(CCCN(C)C(c2occc2C)=O)C)C1 CC1Cc2cc(-c3noc(CSc4nc(Cl)nc(=N)[nH]4)n3)ccc2O1 c1(NC(C=CCNC(c2ccc(CC)o2)=O)=O)cccc2nccn12 N1(CCC=CCC)CCC(C2CCN(C(c3csc([N+](=O)[O-])c3)=O)CC2)C1 C1(CCNC(CN(CC(C)(C)C)C)=O)CC(NC(=O)CC2(C#N)CC2)C1 c1(CN(C2(C3CCCO3)CCCC2)C(=O)C2CC2)ccc(Br)cc1.C1CCC(=O)N1 C(=O)(C(C)(C)C(=O)NC1CC(CCNC(=O)CC2CS(=O)(=O)C2)C1)N(C)C N1(C(C2(C(CC)=O)CC2)=O)CCC(C(=O)NCC2CCC(C)C2)=C(F)C1 N1(C(C(C)SC(C)C)=O)CCOC2(CCN(C(=O)CCn3ccnc3)C2)C1 C1(c2cc(C(=O)OCC)no2)CCCCN1C(=O)C(N)CC1CCS(=O)(=O)N1 CN=c1[nH]c(=NCc2ccc(CN(C)C)cc2F)[nH]c(=NC2CC3C(C2)C3(F)F)[nH]1 C1(NC(=O)C(=O)N(CC(F)F)C2CCC2)CCN(C(=O)CCn2cc(Cl)cn2)C1 N1(C(CCCOCCC)=O)CCCC(CNC(=O)C(c2cccc(C)c2)OC)C1 C1(C)(C(N2CC(c3n(C)ncc3)C2)=O)CN(C(=O)CSCCC#N)C(C)(C)C1 C1(C(N2CC(CC)(CO)C2)=O)CCN(C(C2CC3CCC2C3)=O)CC1 N1(C(C(CC)(C)O)=O)C2CCC1CC(N(C)C(c1csc(C(C)OC)n1)=O)C2 CC(Cc1ccccc1Cl)N=c1nc(N2CC(F)C(F)C2)c2[nH]ccc2[nH]1 CCCC(C)CC(=O)N1CC2C(CNC(c3c[nH]nc3-c3cccs3)=O)C2C1 C1(N(C)C)CCCC(N(C(=O)CCSC(F)(F)F)C(C2CCCCCC2)C2CC2)C1 c1(C(=O)NC(CC)CN(C)C(c2cccnc2S)=O)[nH]c2ccccc2c1Cl N(C1CCc2ccc(Cl)cc21)C(=O)CC1CCCCC1(F)F c1(C(N(CCCCNC(c2nc(CC)oc2C)=O)C)=O)cc2n(c1)CCCC2 c1(C(=O)NCCN(C(=O)CC2CCCC2O)CCC)nocc1Br C1(=O)C(C)CN(C)C(=O)CN2CC(C)(C2)N1C(C)C.C(C)(C(C)C)SC N1(C(C=COC(N2CCC(C(=O)NC)C2)=O)=O)CCC(CC(C)OCC)CC1 c1(C(C(=O)NC2CCC(NC(c3cnoc3C)=O)C2)OC)cccc(Cl)c1 C=CC(C)(C)C(=O)NCc1ccoc1C(N1CC2C(C)C2C1)=O C(c1cc(Cl)cc(Cl)c1)=CC(N1C(C(C)NC(=O)CCCC#N)CCCC1)=O C1(CCC(=O)NC2(C3CC3)CCC2)CCCN(C(C23CCCCC2C3)=O)C1 CC(C)CC(Cn1cc(C2(C)COC2)nn1)NC(=O)CC(C)n1cccc1 N1(C(CCC=C)=O)CCC2CC2(CNC(=O)Cc2cccc3sccc23)CC1 c1(C(c2nnnn2C2CC2)NCC(C)F)cn(-c2ccccc2)cn1 CC1Cn2nccc2CN1C(=O)C(C)(C1CC1)N(C)C(c1ccc(Cl)cn1)=O C(CNC(=O)C(C(C)C)SC)(C(=O)NOCCOCC1CCOCC1)OC CC(O)(CC(=O)NCC1CCCC1NC(C1(c2cccs2)CCCC1)=O)C(F)(F)F C1(CNC(=O)Cn2cncn2)CCC2CN(C(C3(CF)CC3)=O)CCC2C1 N1(C(c2c(CC)ncs2)=O)CCOCC1CC(=O)NCCCc1nc(C)no1 Cc1nc(C(C)C)ccc1NC(N1CCC1c1cn(-c2ncccn2)nn1)=O CCC(C)(C)C(=O)C(=O)N1CCN(CCNC(c2ccc(C3CC3)nc2)=O)CC1 C=C(C)CC(C(=O)NCC(C)(F)CNC(=O)C(O)CSC)OC CC(C)(C)CC(C)(C)C(=O)NC(CNC(c1n[nH]c2c1CC1CC21)=O)C1CCC1 N1(C(COC)=O)CCCC(C)(NC(N2CC(n3cccc3)C2)=O)C1 C1(C(=O)NC(c2cnn[nH]2)(C)C)N(C(=O)CC2CCCNC2=O)CC12CCCC2 C1(C(=O)NCC2CCN2C(=O)CCC2CCOC2)CCCOCC1 Cc1cc(C(N2CC3CC3(CNC(C3(C)CC4CC4C3)=O)C2)=O)nc(C)c1 C(=O)(C#CC1CCCO1)NC1(CC(=O)N(C)CC2CC2(F)F)CCC1 c1(C(N2CCCC(NC(C(CC=C)(C)C)=O)CC2)=O)cccc2ncnn12 N#Cc1cc(F)ccc1C(N1CCC2(CC(NC(C3CCCS3(=O)=O)=O)C2)C1)=O CC(C)CCCCCCNC(C1CCOC1CNC(=O)CN=[N+]=[N-])=O c1(C(N2CC(NC(=O)CC3CCC4CC34)C2)=O)nsc2cc(Br)ccc12 N(C(=NCC(C)SC(F)F)NC(C)C)Cc1nc(-c2ccc(C)cn2)on1 N1(C(C2(C)CC2(Cl)Cl)=O)CCC(C)(NC(c2cncc(NCC(F)F)c2)=O)C1 N1(C(CCCC(C)O)=O)CCCC(C2CCN(C(c3nnn(C)n3)=O)CC2)C1 C1(NC(CCC(N)=O)=O)CN(C(=O)COCC2CCCC2)CC2(CC2)C1 O=C1CCC(CC(=O)NCCc2cc(C(N3CCCC3C(O)CO)=O)no2)CC1 C1(CC)CN(C(=O)CC(C)(C)SC)CCN1C(=O)CCCc1ccccn1 C1(CNC(Cc2nccc(C)c2)=O)CCN(C(c2nccnc2Cl)=O)CC1(F)F C=CC(F)(F)C(=O)NC1(CCCCSC)CC1.C1(=O)C(C)C=CCN1 C(=O)(C(C(=O)OC1(CC(=O)OCC)CCC1)NC(=O)N(C)C)OCC CC(C)(CNC(=O)Cc1cncc(O)c1)CCNC(c1cncc(Br)c1)=O C=CCCN=C(NCC1COC(C)(C)C1)NCC1CCC2(CCCC2)O1 c1(C(=O)NC(C(CO)NC(c2c(OC)nsc2)=O)C)cc2sccc2cn1 C#Cc1cn(C)nc1C(N1CCOCC1CN(C)C(C1C(C)(C)C1(F)F)=O)=O Cc1ccccc1C=CC(=O)NC1CCC(CN(C(=O)C(C)CC2CC2)C)CC1 C1(CNC(C(CC(C)C)(F)F)=O)Cc2ccccc2CN1C(C1CCSC1)=O C(=O)(CC(F)(F)CC(=O)NCC1CCC1NC(C1COCCN1C=O)=O)OC CC1CN(c2ccc(C(N3CC(N4CCOCC4)C3)=O)cn2)CCO1 c1(CCC(=O)NCCOCCN(C(=O)CC)C)ncccc1F.C(N)(=O)COC N1(C(c2cncc(OCC)c2)=O)CCN(C(c2c(CO)n[nH]c2C)=O)CC1C N1(C(CCSC)=O)C2CCC(C(=O)N(C3COCC3(C)C)C)C1CC2 C1(COCC)CCCN(C(C23CC(N(C(=O)C(O)CC)C4CC4)(C2)C3)=O)C1 N1(C(C=CC)=O)CCC(CO)(NC(c2cc(C)co2)=O)C1 C1(NC(CNc2cn(C)nc2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)CC1 c1(C(=O)NCCC(F)(F)F)cc2n(n1)CCCC2.C=C1CNC(=O)CSC1 C1(CC(=O)NC(c2ccccc2)C(=O)NCCC(C)OC)CCCCC1O C1(CN(C(c2ccc(CC)s2)=O)C)COCCN1C(C1CCCN1CC)=O CC1CN(C(C2(C(N)=O)CCC2)=O)CC1CCNC(c1ccnc(C(F)F)c1)=O C1(C(C)CNC(c2cc(Cl)ns2)=O)CCN(C(C2CNC(=O)C2)=O)CC1 c1(C(C(=O)N(C)CC2CCCCN2C(C23CC(C2)C3)=O)O)cc(Cl)cc(Cl)c1 Cc1nocc1C(=O)NC1CC(O)(CNC(c2cccs2)=O)C1 C1(O)(CNC(c2c(C(=O)O)ccc(OC)c2)=O)CCCC12CCOCC2 N1(C(CC(c2cccc(F)c2)C)=O)CCN(C(c2cnc(Cl)s2)=O)CC(O)C1 C(C(CNC(=O)CN1CCCCC1)C(F)(F)F)NC(C1CCOC1)=O c1(C(=O)NC2(CNC(C(C)C3CCCO3)=O)CCCCC2)cncc(O)c1Cl C1(c2c(C)ccnc2)CCN(C(=NCC(C)C)NCC2(C(N)=O)CCCC2)C1 C1(CNC(C2CC=CCO2)=O)CCN(C(=O)CCc2sccc2Br)CC1 N1(C(C(N)=O)=O)CCC(NC(=O)NCC2(Sc3ccccc3)CC2)C(F)C1 c1(CC=C)cccc(C(N2CC(NC(=O)CN(C3CC3)CC)C(C)C2)=O)c1 C#CCCCCCCC(=O)NC1CCC(CCC=C)C1.N12CCCC(CC1)C2=O C#CCC(C)C(=O)NCC(F)CNC(=O)CCc1ccc(C(F)F)cc1 c1(CC)cnc2snnc2c1.C12CN(C(c3ccnc(OC)c3)C)CCN1C2=O C1(OC)CCC12CC(C(=O)NCC1CCCC1NC(c1ccn(C3CC3)n1)=O)C2 C(CCCCC(=O)N1CCSC2CCC12)NC(c1cc(CCC)[nH]n1)=O C1(C(N(CC(CN(C(=O)C=Cc2cnn(C)c2)C)O)C)=O)CCCC2C1C2(F)F CCCCCC(CC)C(=O)NC1CC(CCNC(c2ncccc2F)=O)C1 c1(-c2cc(OC)c(F)nc2)ccc2sc(C(N3CCN(C4CC4)CC3)=O)cc2c1 N1(C(c2c(NC)cnnc2)=O)CCN(C(=O)C(=Cc2ccc(F)cc2)C)C2CC12 Cc1[nH]nc(C(N2CCC(O)(CN(C)C(C3(C)CC=CCC3)=O)C2)=O)c1Cl C1(C(=O)NCC2(OCCNC(C3CC3Cl)=O)CCOCC2)CC2(C1)CC(F)(F)C2 c1(CCC(=O)N2CC(CNC(=O)C(O)CC3CC3)C2)ccc(O)cc1 c1(C(=O)NC2CC(NC(=O)C(F)F)C2)ccc(-c2ccc(Cl)cc2)cc1 c1(CC)nccn1CCN1CCC(NC(=O)CCc2cncs2)C1 CCCC(C(=O)N1CC(O)(CCNC(c2cc(S(N)(=O)=O)cs2)=O)C1)C(C)C C(=O)(CC(C)(C)C(C)(F)F)N1C(C)CC(NC(c2ccc3cncn3c2)=O)C1 N1(C(C2C(CC)CCO2)=O)CCCC(C)(CNC(=O)Cc2ccnn2C)C1 c1(N2CC3(C(NC(C4C(C(C)O)C4)=O)CCS3)C2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CCCC(O)CC(=O)NCc1ccccc1CNC(C1(F)CC=CC1)=O C#CCC(C(=O)N1CC2CC2C1)NC(=O)CC1CC2CCC1O2 C#Cc1cnn(CC(=O)NC2CCCCC2NC(C2CCCN2CC)=O)c1 C1(O)(CNC(c2cc(Br)c[nH]2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1 C1(NC(C2OCCN(C(c3n(CC)ccn3)=O)CC2)=O)C2CCC3C(C2)CC13 c1(OC)ccc(C)c(C(=O)NCC2CN(C(C3CC3OC)=O)CCC2C)c1 N1(C(C)=O)CCN(C(C2(C)CN(Cc3ccc(C)c(Cl)c3)C2)=O)C(C)C1 C(=O)(CCN(OC)C(=O)C1CCCCCN1C)C(C(=O)OC)CC(C)(C)C n1(CCOC)ccc(C(=O)N(C)CC2(C(F)(F)F)CC2)n1.C12CC1CNC2=O C1(NC(C(C2CCC(=O)NC2)C)=O)CCC2CC1CN2C(C1CCC2CC2C1)=O N1(C(C(C(=O)OC)F)=O)CCN(C(=O)C=Cc2cncn2C)CC1C c1(C(=O)NCCN(C(=O)C(Cl)=CCl)C2CCCC2)cccnc1O N1(C(c2ccc(OCF)cc2)C(=O)NC(C(=O)OC)C)CCC(C2CC2)C1 C1(CN(C(c2ccccc2Br)C)C)CCN(C(=O)CC2CCOC2)CC1 c1(C(N(CCN(C)CCc2cn(CC3CC3)nn2)C)=O)nc(Br)n2c1CNCC2 C1(C(N2C(CNC(c3nc(C)n(C)n3)=O)CCCCC2)=O)CC2CCCCN2C1 CC12CC(CC(N3CCCC(C4CCCCN4C(c4ccsc4)=O)C3)=O)(CO1)C2 Cc1cccnc1CC(=O)NCC1CN(C(=O)CC23CCCC2C3)C1 C(c1ccc(O)cc1)=CC(=O)N(CC(C)O)CCNC(C1CN(C(C)C)C1)=O c1(C(=O)NCC(C(C)C)NC(C(CCC)C#N)=O)nc2ncc(C)cn2n1 CCC(Cc1ccccc1)CC(=O)NC1CC(C)(NC(C2CN(C)C2)=O)C1 c1(NC(=O)NC2(c3ccc(Br)cc3)CC(F)(F)C2)cncc(-c2n(CC)nnn2)c1 C1(CNC(c2cnc(C(C)(C)C)[nH]2)=O)C2CCC(C2)N1C(c1ccc(C#N)o1)=O N1(Cc2c(C)noc2C)CCOCC(C(=O)NCC2CC3CCC2C3)C1 c1(C(N2CC3C(NC(=O)Cc4ccsc4)(C3)C2)=O)ccc2cccnc2c1F CC1CN(C(=O)CC2CCCO2)CC1(C)C(=O)NCCN1CCCCC1C c1(N2CCC(CC)(CO)CC2)ncc(S(=O)(=O)N(C)CC2CCOCC2)cc1Cl c1(C(N(CC(C)N(C)C(C2(C)CC2(C)C)=O)C)=O)ccc2c(c1)CCN2C C(=O)(C1CCCc2c(O)cccc21)N1CCCN(C(C2=C(C)OCC2)=O)CC1C c1(CN(S(=O)(=O)Cc2cccnc2)Cc2ccc(OC)cc2)cccc([N+](=O)[O-])c1 N1(C(C2C(C)(C)S(=O)(=O)CC2)=O)CC2CC(NC(c3cc[nH]c3)=O)CC1C2 C1(NC(c2cc(C)nn2C)=O)CCN(C(C2CCC(=O)C(C)C2)=O)CC12CCC2 c1(C(N2CC(C3CN(C(=O)CC45CCCC4C5)C3)C2)=O)ccn2cncc2c1 C1(=CC(=O)NCC2(C)N(C(CCSCCC)=O)CCC2)CN2CCC1CC2 Cc1cc(C(N2CC(c3ccccc3)C2)=O)cc(C)c1.C12(CCSC1)C(=O)N2 CCC(CC(C)C)C(=O)NC12CC1CN(C(=O)C=Cc1nc(C)c(C)[nH]1)C2 C(=O)(CCCC(=O)NC1CN(C(C2CN(CC(C)C)C2)=O)C(C)(COC)C1)NC N1(C(c2ccc(Br)cn2)=O)CC2CN(C(c3ccccc3I)=O)CC2C1 c1(C(N2CC(F)C(F)C2)=O)ccc(-c2cncc(N3CCCC3)c2)cc1F n1(CC)cnnc1C(=O)NC1(CCNC(=O)CC2CC(C)=NO2)CCCC1 C1(CNC(c2c(CC)nco2)=O)(CNC(=O)C(Br)=C(C)C)CC12CCC2 C1(CCNC(c2cocc2C)=O)(NC(C(C2CC2)SC)=O)CCOCC1 C(=O)(C(C(C)C1CC1)N1CCC(CN(C)C)C1)NCCSC C1(C(=O)NCC(C)(CO)NC(c2c(C)noc2C)=O)CCc2ccnn2C1 C12(CNC(CCC=CC)=O)CC1CN(C(c1ccnc(OCC3CC3)c1)=O)C2 CS(=O)CCC(=O)NC1C=CCN(C(c2cc(COC(C)(C)C)on2)=O)C1 C1(C(N2CCC(OC(=O)C3CC3)CC2)C(=O)NC)CC2(C1)CC(C)(C)C2.CC(C)C C1(N(C(c2cc(SC)[nH]n2)=O)CC2CCCCO2)C2CCC1CNC2 C1(NC(c2c(C)n[nH]c2)=O)CN(C(c2c[nH]ccc2=N)=O)CC2(CC2)C1 C=Cc1ccc(C(=O)NC23CC(NC(c4cnn5cc[nH]c45)=O)(C2)C3)cc1 N1(C(C)=O)CCN(C(=O)C(C)(C2CC2)N(C(=O)CCCF)C)CC1 c1(C(N(CC(CNC(C(C)OCCC#C)=O)C)C)=O)oc(C2CC2)nc1C C(=O)(C1=CCCCCC1)NCC1N(C(C(C)=CC2CC2)=O)CC(F)(F)C1 N1(CCn2c(C(C)NCCO)nnn2)C2CCC1CN(CCONC(=O)OC)C2 N1(C(C2CCCN(C)CC2)=O)CC2CCCC1CCC2 C1(CC(=O)NC(C2CCCC2)CC)CCN(C(=O)CC2(C)CCCCC2)C1(C)C c1(CC)cnc(CNC(c2nnnn2CCN2CCOCC2)CCC2CC2C)o1 C(=O)(C1CCS(=O)(=O)c2ccccc21)N(C(CCC=C)c1ccccc1)CC c1(C(C2CC2)NC(=O)NCC2(CC=C)CCCC2)ccccc1Cl c1(CN2CC(NC(c3ccc(Cl)o3)=O)C(O)C2)ccc(F)cc1[N+](=O)[O-] c1(CC)nc(C)c(C(=O)NC2CN(C(C3CC(O)CN3C)=O)CC2O)s1 Cc1cncc(F)c1C(=O)NC1CCC(N(C)C(c2n[nH]c3c2CCC3)=O)C1 c1(C(=O)OC)c(C)[nH]c(C(=O)NCCCN(C(=O)CCc2csc(C)n2)C)c1C c1(C(C)NC(=O)CC2CN(C(=O)CCN3CCOCC3=O)C2)cc(F)c(F)cc1O N1(C(CC(C)O)=O)CCC(C(N2CCCC(c3ccccc3)C2)=O)C(C)(C)C1 N1(CC2(NC(N3CC(OC)C(SC)C3)=O)CCC(C)(C)C2)CC2(COC(=O)N2C)C1 Cc1cc(C(=O)NC2CCC2CNC(c2cn(C(C)C)cc2C)=O)c(C)c(C)c1 c1(C(N(CC(CN(C(C(C)=C(C)C)=O)C)O)C)=O)csc(C(F)(F)F)n1 C(CNC(=O)CSCCC(C)C)(CC(C)C)NC(c1cnc(OC)s1)=O CC(CCNC(c1ccc(-c2cccnc2)cn1)=O)CCNC(=O)C1=CCOC1 c1(C(=O)NC(C)C(=O)NC(c2cc(Br)no2)CO)ccc(Cl)c(Cl)c1 CC1(C)NC(=O)CC1C(N1CCCC(O)(CCNC(C2(S(C)(=O)=O)CC2)=O)C1)=O c1(C(=O)NCC(C)(O)CNC(=O)CNC(=O)C2CC2)cc(C(F)(F)F)cc(F)c1 C(=O)(CC(C)(C(F)(F)F)Nc1cc(OC(F)F)c(O)c(F)c1)OC C(CCCC(=O)NC(C)CCC1CCCO1)N(C(C(SC)SC)=O)C C1(NC(C(CC)C)=O)CCC2(CCN(C(=O)CCCCN(C)C(C)=O)CC2)C1 CC(C)CCC(C(=O)N1CCC1C)NC(c1cccc(CC#N)c1)=O c1(-c2cn(CC)nc2C(F)(F)F)cnc2ncc(C(=O)NCC(C)OC)n2c1 c1(C(N2CCCC2CO)=O)nnc2ccc(-c3cnccn3)cn12 S(=O)(=O)(c1cccc(C(=O)NC2C(NCC)CC2)c1)NC(=O)C(C)NS(C)(=O)=O N1(C(C(C)(C)OCCC)=O)CC2(C)CC1(C(=O)NCc1ncc(C)cn1)C2 N1(C(c2c(CC)non2)=O)CCCC(CO)(NC(=O)C(F)C(C)C)C1 Cn1c(I)cc2c(N3CCc4sc(-c5cnc6sccc6c5)nc4C3)ncnc12 N1(C(CC(=O)NC)=O)CCCC2(NC(C34COC(CCO3)C4)=O)CC2C1 C1(C(N(C)Cc2noc(=O)n2C)=O)CCN(C(C2C3CCCC23)=O)C12CCC2 CCCC(CC)C(=O)NCc1ncoc1C1CN(C(c2[nH]ccc2C2CC2)=O)C1 c1(C(N2C(C(C)NC(c3[nH]ncc3C#N)=O)CCCC2)=O)ccc2c(c1)OCC2 c1(CC(N2C(CNC(c3c(COC)nn[nH]3)=O)CC2)=O)ccc(Cl)cc1Cl c1(CN(C(c2cccc(C)c2)C)C)cc(F)ccc1O c1(C(=O)NCC2CCN(C(COCCCC#C)=O)CC2)cccc2c1C(=O)NC2 c1(CC(N2CCC3CN(C(=O)C(F)CC4CC4)CC23)=O)ccc([N+](=O)[O-])cc1Cl C1(NC(C(C)=CC)=O)CC2(C1)CN(C(=O)C(C)SCC1CCCO1)C2 N(C1c2ccccc2CC1C)C(C(=O)NCc1cc2cc(C)ncc2cc1)=O C(=O)(C1=CC2CCCCC12)N1CCC(N(C(=O)CC2CCNC(=O)C2)CC)CC1 N1(C(C=CC(=O)OCCCC)=O)CCCC(F)(C(N2CCSCC2C)=O)C1 Cc1c(N)ccc(C(=O)NCCC2CCC(NC(=O)C(C)(C)C(C)(F)F)C2)c1F c1(C2C(=O)N2)ccc(OCC(F)F)cc1.CCC(C)(C)OCN1CCCC1 c1(-c2cc(C(=O)NC3C(NC(C(CSC)O)=O)CC3)on2)ccc(C)cc1 c1(N2CCC(C)(F)C2)cccc(S(=O)(=O)N2CCCC(OCCO)C2)n1 N1(C(C2(CCCC)CCC2)=O)CCCC(CNC(c2cc[n+]([O-])cc2)=O)CC1 c1(C(=O)NCCCN(C(=O)CC2CCCC2C)CC)cccnn1 Cc1cc(Cl)ccc1C(N1CC(CNC(c2c(C)nnn2C(C)C)=O)C(C)C1)=O S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1C2CC(NC(=O)Cc3cnc[nH]3)CC1CC2 CC1(C)CC(NC(c2cnn[nH]2)=O)CN(C(=O)C(=Cc2c[nH]cn2)F)C1 c1(NC2C=CCC(C3CCCO3)C2)ncnc2cc(C3CC3)nn12 C(=O)(CC(C)C(C)(C)NC(=O)C(C)c1cc[nH]n1)Nc1c(CC)nc(C)cc1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)CC(C)C)C(C#N)C1 N1(C(C(CNC(C(CCOC)C)=O)(F)C(C)C)=O)CCCC2C(=O)NCC12 C1(C(=O)NCC2CCCN(C(C(C)O)=O)C2)CNc2ccccc2O1 O=C(CCCNC(c1cccnc1)=O)NC1CC1CNC(C1CC(CF)C1)=O CC1(C)CC(C(N2CCCC(F)(CNC(C3CCC3)=O)C2)=O)CC(C)(C)C1 N1(C(=O)NC(c2ncsc2Br)C)CCC(F)(F)C(S(C)(=O)=O)C1 N=c1ncc(C(=O)NCC2CN(C(=O)CC3CCCCCO3)CCO2)c[nH]1 N1(C(C2(C)C(C)CN(C(=O)CC3C=NN(C)C3=O)C2)=O)Cc2cccnc2C1 C(=O)(C1=CCCSC1)NC(C(=O)NC1CCN(CC)CC1)Cn1cncn1 c1(C(=O)NC2CCN(C(C(CC)(C#N)CC)=O)CC2O)cccc(P(C)(C)=O)c1 C1(C)(C(N(C(CCC)C)CC)=O)CCCN(Cc2ccc(N)c(Cl)c2)C1 c1(C(C)=O)cc(CCC(=O)NCC2CC(NC(=O)C=CC3CCCCC3)C2)oc1C c1(C(N2C3CC(NC(C(c4ccccc4)C)=O)C3CC2)=O)cc(Cl)c(F)c(Cl)c1 N1(C(CC(=O)NCC)=O)CCC(C(N2CCC2(C)C)=O)(CC)C1 C#CCCCC(C)C(=O)N1CCN(C(=O)C#CC2(CC)CC2)CC1CC(F)F CC(C)(C)CCC(=O)N1CCOC(CNC(c2n[nH]cc2F)=O)C1 CC(C)C(C)(CNC(=O)C#CC1CC1)NC(=O)Cc1ccc(-n2ccnc2)cc1 C(=O)(C(C)(O)C(F)(F)F)NC1CCN(C(c2c(OCC)nc(C)cc2)=O)C1 c1(OC)ccc(CN2CC3CC2C3C(N2CCC(N(C)C)CC2)=O)c(F)c1F C=CCC(C)C(=O)NCCCCC1(NC(C2CC(C#N)C2)=O)CC1 CC1CCC(C(=O)NCc2cc(O)nn2C)N(C(C2CCN(C(N)=O)C2)=O)C1 N1(C(C(CCOC)NC)=O)C(C(=O)Nc2cccnc2OC(C)C)C2CCCC12 CC1(C)CC(O)CCN(C(=O)C(F)CC(C)(C)NC(=O)CC2CCCO2)C1 C1(NC(Cn2c(C)nc(C)n2)=O)C(C)CCN(C(=O)COc2cccnc2)C1C c1(C(=O)NCC(CN(C(=O)C(F)CC2CCCC2)C)O)noc2c1CCCC2 c1(C(N2C(CCNC(C3(C)C(C)C3)=O)CSCC2)=O)cc2ccc(Cl)cn2c1 C1(C(=O)NC(CC)CO)CC(N=[N+]=[N-])CN1C(c1cc2occc2[nH]1)=O c1(C(N2C(C(=O)NCc3nc(CC(=O)NC)cs3)C=CC2)C)ccnc(CO)n1 c1(C(c2n(CCCC)nnn2)NCc2nc(CC)no2)cc2nc(F)ccc2o1 c1(C(N2CCC3CCC(NC(COC(C)C)=O)C32)=O)ccc(O)c2ncccc12 C1(NC(C2CCC(CC)CC2)=O)CC(CNC(c2nnn(C)c2C)=O)C12CCC2 C(CS(=O)(=O)CC(=O)NCC(C1CCCC1)NC(=O)C(C)O)OC C(CCN(C(=O)C(C(C)C)NS(N)(=O)=O)C)(C(C)C)NC(Cc1nc(C)sc1)=O C1(CNC(C(=O)NC(c2ncnn2C)C)=O)CCC2(CCCC2)O1 CCS(=O)(=O)NC(C)C(=O)NC1CC(NC(C2CC2C(=O)OC(C)(C)C)=O)C1 n1(CC(N2C(CNC(COC)=O)C=CC2)=O)c(C(C)(C)C)nc2ccccc12 CC1CCCN(C(=O)C(Cc2ccoc2)NC(c2ncn3c2CCC3)=O)CC1 c1(OC)nc(C)ncc1C(=O)NCC1CN(C(=O)CCc2cn(C)nn2)C1 c1(CN(c2n(CCC#C)c(CCCS(N)(=O)=O)nn2)C)ccc([N+](=O)[O-])cc1 c1(CSC)c(NC(N2CC(N(C)C)C(c3cn(CC(C)C)nn3)C2)=O)c[nH]c1C N1(C(CC)=O)CCC(C(F)CNC(C2CCCN2C)=O)CC1 C1(N(C)C)C2CN(C(=O)Cn3cc(C(c4ccc(F)cc4)(F)F)nn3)CC12 c1(CNC(=O)C(=O)NCC2CCCC23CC3)ccccc1-c1ccccc1 CC1CCC(F)(C(=O)NCc2ccccc2CN(C)C(c2c[nH]c(=N)s2)=O)CC1 C1(CC)(CC)CC(NC(=O)C(C)COC)CN1C(=O)CC(C)(C)SC CC1C(=O)NC(=O)CN1C(=O)CC12CCN(C(=O)CCCc3ncco3)CC1C2 C1(C(N(C)CC2(O)CCOC2)=O)CN(C(=O)CCS(C)(=O)=O)CC(C)(C)C1 c1(N2CCC(OCCNC(CC=C)=O)C2)ncnc2sc3c(C)cccc3c12 N1(C(C2C(NC(C3N(C)CC4(CC4)C3)=O)COC2)=O)CCC12CCSCC2 c1(C(=O)OC)ccc(C(N2CCC(N(C(=O)C(C)N(C)C)C)C2)=O)c(F)c1 CC1CN(C(=O)C=CC2CCCN2C)CCN1C(=O)C(N)=O n1(CCC(=O)NCC(C)(CO)NC(C(n2ncc(C)c2)C)=O)ncn(C)c1=O c1(C(=O)NCCCNC(=O)CNC(c2ccco2)=O)ncc(Cl)cc1F C(c1ccc(C)cc1C)=CC(=O)NC1CCC(CCNC(C(CC#C)C)=O)C1 C1(NC(C2(C)CCC(C)CC2)=O)CCC2CC1CN2C(c1ncnc(O)c1Br)=O C1(CN(C(=O)Cc2nc[nH]n2)C)CC(NC(C2CN(C(N)=O)C2)=O)C12CCC2 c1(C(=O)NCC2C3CN(C(C4CCN(CC5CC5)C4)=O)CC23)cccc(Cl)c1F c1(C(C)C)cccc(C(N2CCC(CNC(=O)C(C)(C)c3cncnc3)C2)=O)c1 Cn1ncc(N)c1C(=O)NCCCN(C(=O)C(C1CCCO1)C1CC1)C1CC1 c1(N2CC(NC(=O)NCC3C(C(=O)OC)CCO3)C2)ccc(F)cc1F C(CCS(C)(=O)=O)(C(=O)Nc1csc(SCCN2CCN(C)CC2)n1)OC N1(C(C2CCC(CC)O2)=O)CC(NC(=O)COc2cccc(F)c2)C(C)C1 CC(C(=O)N1CCCC(CN(C(=O)Cn2nnnc2C2CC2)C)C1)P(C)(C)=O C1(C(=O)NC(C2N(C(CCC=CC(C)C)=O)CCC2)C)CC(C2CC2)=NO1 c1(C(N2CCCC(C)(CNC(C3(CO)CC3)=O)C2)=O)c(F)ccc2n[nH]cc12 C1(C(=O)NC(C)CCc2cn[nH]c2)CN(C(=O)OC(C)(C)C)CCC1(C)C C1(C)(C(N2CC3C(NC(c4c(COC)ncs4)=O)C3C2)=O)CCC2CC2C1 C#Cc1ccc(C(=O)NCC2CCC(NC(=O)CC3CCC3)C2)nc1 N1(Cc2c(OC)ccc(Br)c2)CC2C(C1C(=O)NCCC(F)(F)F)C2(C)C C=CC1(CC(=O)NCCCCN(C)C(C2CCCC(C)CC2)=O)CCCCC1 C1(CNC(c2ccc(CO)c(F)c2)=O)CC2CCC1N(C(=O)Cc1cscn1)C2 c1(OCC)ccc(CCC(=O)NCC2CCN2C(C2CC(F)C2)=O)cc1 c1(CNC(C2(CNC(C(C)n3cncn3)=O)CCC2)=O)ccc(F)cn1 N1(C(C2(C)CC(O)CN2C(C2CCC2C#N)=O)=O)CCC2(CNC(=O)C2)C1 C(=O)(NNc1ccc([N+](=O)[O-])cc1)c1c[nH]c(=NCCC2CC(C)(C)OC2(C)C)s1 Cc1ccc(F)c(C(=O)NCC2CN(C(c3cc(C(C)(C)C)no3)=O)CCO2)c1 c1(C(N2CC(NC(C(C)(C)c3cnsc3)=O)C(CO)C2)=O)ccn2ccnc2n1 C#CCCCCCC(=O)N1CCCC(C(=O)NCCc2cccc(O)n2)C1C c1(OC)ncc(C(=O)NC2CC(NC(=O)CC(C)(C)O)C2)cn1 Cc1ccc(S(=O)(=O)N2CCC(C(N3CCCCC3C(=O)N(C)C)=O)CC2)cc1C CN1CCN(C(=O)CC2CCOC2(C)C)C(CNC(=O)CSCC(F)F)C1 c1(C(=O)NC(C2CCN(C(c3ccc(Cl)s3)=O)C2)C)cnc(O)c(F)c1 CC1(O)CC(C(=O)NC(C2CCCCC2)CNC(C2CCO2)=O)C1 N1(C(Cc2cc(C)cc(F)c2)=O)CCC2CN(C(c3n[nH]cc3C)=O)CC12 C(=O)(CCC(F)(F)F)NC1(C(N(C)CCc2cccnc2)=O)CCC1 N1(C(c2cn(C)nc2C(C)(C)C)=O)C2CCC1C(NC(=O)C1CC1)C2 c1(-c2cn(C3CN(C(CC4(OC)CCC4)=O)C3)nn2)cc2ccccc2s1 Cc1cnn(C(C)C)c1C(=O)NCC1CN(C(C2CCCC2C(F)F)=O)CC1O Cc1nn(C)c(C)c1C(=O)NCC1COCC1NC(=O)Cc1cc(F)ccc1O n1(CC)cnc2[nH]c(=NC3CCN(C4CC4)C3)nc(N3CCC(OCC)C3)c12 c1(C(=O)NCC2CN(C(CCc3cc(C)no3)=O)C(C)C2)ccc(Cl)c(N)c1 C1(NC(=O)Cc2cc(C(=O)O)nn2-c2ccc(F)cc2)CC(C2CCC2)C1 C1(NC(=O)C=CCF)(CO)CCCN(C(=O)Cn2cnc(-c3ccccc3)n2)C1 c1(C(N(C(C)C(=O)NC2CN(C(=O)OC(C)(C)C)C2)C)=O)nc(O)n[nH]1 c1(OC)cc(CNC(N2CCC(N3CC=CCC3)C2)=O)cc(C)n1 C=CCCCC(C)(C)C(=O)N(CCNC(c1ccc(COC)cc1)=O)C1CC1.C1(CC)CC1 c1(C(N2CC3(CCCN(C(C4N=C(C)SC4)=O)C3)C2)=O)ncn2c(C)cc(C)nc12 Cc1cc(C)c(NC(C2CCN(C(=O)C(N)CN)CC2O)=O)cc1Br C1(CNC(c2n(CCOC)nnn2)c2cnc(Cl)s2)CC2CC1CC2O C1(NC(=O)C2=C(Cl)CC2)CC2CC1CN2C(c1cc(C(F)F)ccc1Cl)=O N1(C(c2cnccn2)C(=O)Nc2ccccc2)CC2CC(F)(F)C2C1 C1(c2nnnn2CCCSC)(NCc2cnc(CC)o2)CCOCC1C C1(CC)CN(C(=O)CC2OCCO2)CC1C(=O)NCC(C)(O)C(F)F CCCC(O)C(=O)NC1(CCOC)CCN(C(c2ccnc(C3CC3)c2)=O)C1 CCCC(CNC(=O)Cc1cnc(C)[nH]1)NC(=O)CCN1CCCC1=O CC1CCc2nc(N3CCC(Nc4ncccc4[N+](=O)[O-])C3)c(C#N)cc2C1 S(=O)(=O)(c1cc(Br)cc(Cl)c1O)NC(c1c(OC)cc(C)cc1)C1CC1 C1(NC(c2c(N(C)C)cccn2)=O)CN(C(C2CC2(C)C)=O)CC(F)(F)C1 C#CCC(C)(C(=O)NC1CN(C)C(=O)C1C)NC(=O)COCCF N1(C(=O)CSc2ccc(Cl)cc2)CC2CN(C(c3cnco3)NCCO)CC2C1 C12CCCC1C(=O)N2.C1(COCC)(NC(=O)C2CC2)CCC1 CCC(CC(=O)N1CCN(C(C2OCCC2(C)C)=O)C(CCO)C1)C(F)F c1(C(=O)NCCNC(N2C(C)(C)C(O)CC2)=O)c[nH]c2cnccc12 C=CC1CC(N=c2nc(N3CCCC(S(N)(=O)=O)C3)cc(C(F)(F)F)[nH]2)CCO1 C1(NC(COCC(=O)NC)=O)CCCOC12CCN(C(=O)CC(C)N(C)C)CC2 N1(C(C2(CC#C)CC2)=O)C2CCC1CC(NC(c1csc(C)c1C)=O)C2 C1(NC(CC2CC(SC)C2)=O)CC2(C1)CC2NC(c1cc(C)no1)=O Cc1cnn(C)c1CC(=O)NC1CN(C(c2coc(C(F)F)c2)=O)CC1O N1(C(C2(C(=O)NC)CC2)=O)CCN(C(=O)CN(C(=O)C(C)C)C)CC1C.C1CS1 N1(C(CNC(C)=O)=O)CCCC(CO)(CNC(c2cc(Cl)n[nH]2)=O)C1 c1(N(CC(C(C2CC2)OC)(F)F)C)ncc(C)cc1Br C12(C(N(CCNC(=O)Cc3cccn3C)CC)=O)CCCC1OCC2 C1(N(C(C(C)OC)=O)C)CN(C(c2cccc(-c3noc(C)n3)c2)=O)CC1(C)C C1(O)(CC(C)NC(CN(CC=C)C(C2(OC)CC2)=O)=O)CCC1 C(=O)(C1=CCCCC1C)NC(C1CCC1)CNC(C1(OC)CC1)=O c1(NC)cnc(C(=O)NC2CCCC2CNC(C2(C(N)=O)CCC2)=O)cn1 C1(C(N(CCOC)CCNC(=O)CCSn2ccnn2)=O)CCC2(CCC2)C1 c1(CC)[nH]nc(Cl)c1C(=O)NCCN(C(=O)C(CC1CCCO1)OC)C c1(CCC(=O)N(C)CC2N(C(C(C(C)C)SC)=O)CCC2)cccc2c1OCO2 CC1(C)CC(=O)CCC1C(N1CC2CCC1CN2C(=O)CC1CC=CC1)=O S(=O)(=O)(c1c[nH]c(C(=O)O)c1)NC(C1CCN(c2ccccc2Cl)C1)=O c1(C(C(=O)NC2CCC2)N(C)CC2CCCCC2O)n[nH]c2c(F)cccc12 N1(C(c2ccc(CC)cc2C)C(=O)NCC(F)F)CCCCCCC1C C1(C(C(=O)N(CC(=O)NC2CC2CSC(F)F)C2CC2)O)CCCCC1 C1(CC(=O)NCCCN(C(=O)CC(C)n2cccn2)C(C)C)CCCCC(=O)N1 C1(CNC(Cc2cc(C)on2)=O)CCN(C(c2cc(Br)c(C)o2)=O)CC1 C(=O)(C1=NOC(C)C1C)NC(CC=C)CNC(c1csc2nnsc12)=O C1(CC)CCC(C)CN1C(C1(CNC(=O)Cc2cc[nH]c2)CC(C)(C)C1)=O C(=O)(CCCCCCc1ccccc1)NCC(CCOC)NC(=O)C(C)CSC C1(O)(CN(CCC(N2CCC(COC)C2)=O)C)CCCCC1 C=CCCCC(C)(C)C(=O)N1CC(C2(NC(=O)CNC(C3CC3C)=O)CC2)C1 C(=O)(C(F)CC(C)C)N1CCC(CCNC(CCN2CCN(CC)CC2)=O)C1 C1(NC(C=COCC)=O)CN(C(C2CCOC2(C)C)=O)CCC1CO C1(CC(=O)NCCC2(C(=O)NCc3c(C)ccs3)CCCC2)CC(=O)NC1=O Cc1onc(C(=O)NC(CNC(C2(F)CC2C)=O)C2CC2)c1Br C(=O)(C(C(C)(C)C)N(C)C)N1C(CCNC(c2c(C(C)C)cco2)=O)CCC1 N1(C(CCc2cc(OC)no2)=O)CCN(C(c2cnc(O)s2)=O)C(C)C1 CC(C)C(O)C(C)(C)C(=O)NC1CN(C(=O)C=CCN2CCCCC2)CC1C C(=O)(C1COc2ccc(F)cc21)N1CC(O)(C(C)NC(=O)Cc2ccoc2)C1 c1(CC(=O)NCCN(C(=O)CC2CCC2(C)C)CC)ccccc1C N1(C(C(N)=O)=O)CCC(O)(CCNC(=O)CNC(=O)CC2CCCCC2)C1 Cc1ccc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)C2C)c(C)n1 CCC(C)C(O)C(=O)N1CC(C(C)(C)O)(CNC(=O)CCc2ccco2)C1 Cc1cc(C(=O)NC23CC(CO2)N(C(=O)CC2C(=O)NN=C2C)C3)c(C)c(C)c1 c1(C(N2CC3CN(C(c4cc(Br)ncc4Cl)=O)C3C2)=O)ccc(Cl)c(Cl)n1 CCC(O)C(=O)N1CCC(C(C)(C)NC(=O)CCCn2ccnc2C)C1 Cc1nnc2n1CCC2(C)C(=O)N1CC(NC(c2ccc(C#N)[nH]2)=O)C(F)C1 Cc1ccc(OCC(=O)NC(C(=O)NCc2[nH]nnc2C)c2cccs2)c(C)c1 C1(C(C(=O)NCCC(=O)N2CCC2CF)F)CCOCC1 c1(C(N2CC(F)C2)=O)cc(N2CCOC(c3cccc(F)c3)C2)ccn1 CC1OCCN(C(=O)CC2(C)CCN(C(c3cc(Cl)no3)=O)C2)C1 C12(CC(CO)C1)C(=O)N2.c1(CC(=O)NCCCC2CCOC2)ccc[nH]1 Cc1cc(CN2CCCCC2CNC(=O)Cn2cccn2)ccc1C(F)(F)F N1(C(CC2N(C(COC3(C)CCC3)=O)C3C2CCC3)=O)CC2CC(O)CC2C1 Cc1cc(Oc2ccccc2CC(F)(F)F)ccn1.N1(C2=CCCC2)C(=O)N1 c1(C(N(C2CN(C(=O)C(C)CSC)C2)CC)=O)ccc(C(F)(F)F)cc1 C(=O)(CC(C)C(C)(C)NC(=O)CN(C)C(=O)OC)N1CCC(O)(CCC)CC1 c1(CN(c2n(C)c(C3(O)CCCC3(C)C)nn2)C2CCC2)ccc(P(C)(C)=O)s1 C12(CC(=O)N)COC(C(=O)Nc3cccc(CO)c3)(C1)C2.C(=O)(C1CC1)NCCO c1(C(N2C(C)CCC(NC(=O)C(F)(F)CC3CC3)C2)=O)ccc2oc(O)nc2n1 CC1C(NC(c2ccc(O)cc2)=O)C(C)CCN1C(=O)CC1CCCC(C)C1 CCC(C)(C(=O)NC(C(=O)NCc1ccnc(OC)c1)C(C)C)OC Cc1ncn(C)c(=O)c1C(=O)NCC(C)(C)NC(C1CC(C)N(C)C1)=O C1(CNC(C2CC=CCN2C(c2cc(Cl)n[nH]2)=O)=O)(CO)CC2CC2C1 CC(C)CC(O)C(=O)NC1CCCC1N1CCN(C(c2occc2Cl)=O)CC1 CC(C)C(C#N)C(=O)NCC=CC(=O)NC(c1ccco1)C N1(C(CCC)=O)CCCC(C)(NC(c2ccnc(OC)c2F)=O)C1 C(c1cc(F)c(F)c(F)c1)=CC(=O)NCC1CC(CNC(C2CC(O)C2)=O)CO1 C1(C(=O)NC2CC3(CN(C(C=C4CCN(C)CC4)=O)C3)C2)CCn2nnnc2C1 C(C1CCCCCC1)=CC(=O)NC1(CN(C(=O)CC2CCCC23CC3)C)CC1 C1(C(=O)NCC2CC(NC(c3sccc3C(F)F)=O)C2)COCCO1 C(=O)(C(CC)CC(F)(F)F)NC(C1(O)CCN(C(C(C=C)(C)O)=O)C1)C CN(C(=NCC1CC1)NC1CCCOCC1)CC(c1ccc(F)cc1F)(F)F N1(C(CCc2n(C)ncc2)=O)CCC(NC(=O)C(F)=CCCF)CC1C1CC1 c1(C(=O)NC23C(CN(C(C4CCN(C(C)=O)C4)=O)C2)C3)ccc2n[nH]c(C)c2c1 c1(CCC(=O)NC23C(CN(C(C(C)OC)=O)C2)C3)cc(F)cc(F)c1 c1(CNC(CC(C)(C)C)=O)c[nH]c2cccc(Cl)c12.N12CCN(CC1)CCC2 c1(CN(C(CNC(c2ccccn2)COC)=O)C2CC2)scnc1C C1(C(N(CCSC)CC)=O)CC(C)CCN1C(c1cc(C)[nH]c1C)=O N1(C(Cn2ncc(C#C)c2)=O)CC2(C(=O)Nc3ccc(F)c(COC)c3)CC1CCO2 N1(C(C(C2CCCC2)OC)=O)CCOCC(CNC(C2CCCC(C#N)C2)=O)C1 C1(C(=O)NCCCNC(C(C(C)C)Cc2ccccc2)=O)COCC2(CCC2)O1 C(=O)(C(O)C(F)(F)F)NCC(CC(=O)NC(c1ccccn1)CO)O c1(C(N2CCC(C(C)C(=O)NC3CC4(CCC4)C3)C2)=O)ccc2ccoc2c1 C(CO)(C(C)(C)CO)NC(C(C)(C1CCC1)NC(C1CN(C)C1)=O)=O C1(C(N(CCN(C(C(C)=C(CC)C)=O)C(C)C)C)=O)CCCCC1F c1(C(N(C(C)C)CCN(C(=O)CC2(C)OCCO2)C)=O)ccc2nc(O)[nH]c2c1 C1(C(=O)NCCCC(CCC)NC(=O)CCCC(N)=O)CCS(=O)(=O)C1(C)C CC1(C)C(C(N2CC(F)CC2CNC(C2(O)CCOCC2)=O)=O)CCS1(=O)=O C=CCC(CC(C)C)C(=O)NC1CCCC1NC(c1cnc(C(=O)OC)s1)=O C1(NC(C(C#C)(C)C)=O)CN(C(C2CC23CCOCC3)=O)C2(CCOCC2)C1 C1(NC(Cc2cn(C)nc2)=O)CC(CC(=O)NC2CC(C)(C(N)=O)C2)C1(C)C C(=O)(CC(F)(F)C(F)F)NC(CNC(c1ccc(CC)cc1N)=O)(C)CC(C)C n1(CC)nnc(C(=O)NCC2CC(C)N(C(=O)CC(OCC)OCC)C2)c1C C1(CC(=O)N(CC(C)N(C)C(c2cc(C(F)F)ncn2)=O)C)SC(=N)NC1=O C(=O)(CC1=CCOCC1)NCC1N(C(CC(C=C)(C)C)=O)CCCC1C C1(CNC(Cc2c(C)noc2C)=O)N(C(=O)CC2CCC(=O)O2)CCC1(C)C c1(C(=O)NC(C(C)NC(c2ncc(OC)nc2)=O)C)c(F)cccc1Br c1(Cc2scc(C(N(C3CCN(CC(F)F)C3)CC)=O)c2)ccccc1 Cc1csc2ncnc(N3CCN(C(c4nn(C)c5ccccc45)=O)C4CC34)c12 c1(C(=O)NCC2CSCCO2)cc(C(F)F)[nH]n1 C1(NC(c2n(C=C)ncc2)=O)CC2CCC1N(C(=O)CCCC#CC)C2 c1(C(N(C2CCN(C(=O)CCc3ccoc3)C2)C)=O)ccc(CO)c(Cl)c1 N1(C(C=C(C)C(C)(C)C)=O)CCC(C)C(N(C)C(C2CCC3(CCC3)O2)=O)C1 c1(C(N(C(C)CNC(=O)Cc2cnccc2Cl)C)=O)cc2n(n1)CCN(C)C2 C1(OC)CC(NC(=O)C(F)(F)C(F)F)CN(C(=O)CC(O)c2ccccc2)C1 Cc1cc(CN2CC(N3CCN(S(=O)(=O)CC4CCC4)CC3)C2)c(C)[nH]1 C(=O)(CC(O)CN(C)C)NC(C)CCNC(=O)CC1(C)CCCO1 Cc1ccc(C(=O)NCC2CN(C(=O)CSCC(N)=O)CCO2)c(N)c1 c1(CC(=O)NC(CC(C)C)CNC(c2cnn(CCF)c2)=O)ccc(Cl)cc1Cl O=C1CCCCC(C(=O)NCCC2CN(C(c3ccncc3)=O)C2)N1 C(=O)(CS(=O)(=O)N1CCOCC1)NCCCOCCN(C(=O)C(C)(C)F)C S(=O)(=O)(c1ccc(Br)s1)NC(C1N(C(c2cccc(C)c2)=O)CC2(CC2)C1)=O C(C)(CCCCCO)NC(C1(CNC(=O)COC2CCCC2)CC(=C)C1)=O c1(CN(C(=O)C#CC2CC2)CCNC(COCC#C)=O)ccc(OC)cc1 N1(C(C(CSC)OC)=O)CCCC(O)(CNC(c2ncnc(C)c2C)=O)CC1 Cn1c(C(=O)NC2CC2NC(c2csc3ccccc23)=O)cc2sccc12 N1(C(CCCCCNC(N)=O)=O)CC(NC(C2CC(F)(F)C2)=O)C(C2CC2)C1 c1(C(N(CC)CC2CCCN(C(=O)Cc3csnc3C)C2)=O)nn(C)c(N)c1C C1(C(N(C2CCN(C(c3sccc3-n3ccnn3)=O)C2)C)=O)CCC(O)C1 c1(NC=O)c[nH]c(=NCCc2ccc(O)nc2)o1.C(C)(C)(C)N(CC=C)CC=C Cn1nnc2cncc(C(=O)NC(C)(C)CNC(C34CCC(C3)C4)=O)c12 C1(c2nnnn2C(C)C)(NC(c2ccccc2Br)CC)CC(C)SC(C)C1 c1(C(=O)NC2(CCNC(C34CC(C)C3C4)=O)CCC2)cccc2sncc12 N1(C(CC(=O)C=O)=O)CCN(C(=O)CCc2nc[nH]n2)C2CCCCC12.CNC c1(C(=O)NC2CCCN(C(CCCC#C)=O)C2)ccc(F)cc1C Cc1cc(Cl)nc(C(N2CCC=CCC2)=O)n1 c1(OC)ccc2[nH]c(C)c(C(=O)NC(CNc3ncccn3)CO)c2c1 c1(CCCOC)ccc(C(N2CC(NC(=O)C(O)CSC)C(O)C2)=O)c(O)n1 C(C)(C(=O)C(C1CCCC1)NC(=O)NCCl)(N(C)C)C1CC1.c1(O)ccncc1.C1C(=O)N1 c1(C(=O)NCC2(NC(CSCC=C)=O)CC2)coc(CN)n1.c1ccccc1.C1(S)CC1 C1(CNC(C(C(C)(C)C)(C)C)=O)CC2(CCN(C(C3CCNC3=O)=O)CC2)CO1 N1(C(C(C)NC(c2cccs2)=O)=O)CCCC(NC(C2(CO)CC(C)(C)C2)=O)C1 Cc1cccc(C(=O)NC(C)(C)C(C)NC(c2ccc(Cl)s2)=O)c1F N1(C(CCc2ccc(C)nc2)=O)CCN(C(c2cc(C)no2)=O)C2CCC12 N1(C(c2cn3cc(C)nc3cc2)=O)CCC(C2CCN(C(=O)C(C)O)CC2)CC1 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)CC(CC(=O)OC)C c1(SC)ccc(C(N2CCC2CNC(C2CC(O)C2c2ccccc2)=O)=O)o1 Cc1ccc(C(C)C(=O)NCCC2CC(NC(C3CC(OC)C3)=O)C2)s1 C(=O)(C1CCCn2cnnc21)N(CCCN(C(c1cncc(SCC)n1)=O)C)C N1(C(CCC(C)=O)=O)CCCC2(NC(C3CC(=O)N3)=O)CCCC12 c1(N2CCCC(C(N)=O)C2)nccc(=NCc2ncc(Br)s2)[nH]1 c1(-c2ccn(-c3nnc(CCSCC)o3)n2)c(F)cccc1F CCC(C)(C#N)C(=O)NC1CC(C(=O)NCCC(C)(C)C2CC2)C12CCC2 Cc1c(CC(N2CCCC2C2(NC(=O)C(C)SC(C)(C)C)CC2)=O)cnn1C Cn1cc(C(=O)NCCCS(=O)(=O)N2CCCC2)c(Br)n1 c1(C(=O)NCC(C)NC(=O)C(N2CCOCC2)C2CC2)ncoc1C1CC1 C1(C(N(CC(=O)NC)CC=C)=O)CCOCC1NC(c1cccc(=O)o1)=O N1(C(C2C(C)C2C)=O)CCC2(C1)CN(C(C1CCC(C)(C)O1)=O)C2 c1(OC)ccc(C)c(OC)c1C(N1CC(NC(C2(O)CCC2)=O)CC(F)C1)=O C(=O)(C(CC(C)CC)NC(=O)CCc1cnccn1)NC(CC#CC)CO C12(CNC(CNC(C(C)SCC)=O)C(C)C)CCCC(CO1)C2 C1(CS(C)(=O)=O)CN(C(c2ccccc2F)=O)CCN1C(C1COCCO1)=O c1(OC)ccsc1S(=O)(=O)NCC1(c2ccccc2F)CC(OC)C1 CC1(C)CC(N(C(=O)CC2(C)CCN2C(C2(O)CCSCC2)=O)CCO)C(C)(C)O1 C1(CC(=O)N(C2CCCNC2)C2CC2)CNC2CCCCC12 C(=O)(C1=NOC(CNC(=O)Cn2cncn2)C1)N1C(CSC)CCC1 C1(C(=O)NCC(N2CCCCC2)=O)CN(C(=O)Cc2cncnc2)CCO1 c1(C(N2CCCC(CNC(C=NOC)=O)C2)=O)c(OC)cc(OC)c(OC)c1N CC(CN(C)C)CCC(=O)NCC1CC(O)CN1C(=O)Cc1ccnc(Cl)c1F C(=O)(N1CCC(C(=O)N(CC(F)F)CCO)O1)c1c(C)nc(C)o1 C1(C(=O)NCCc2ccc(Br)s2)COCCN1Cc1cccc(O)c1 N1(C(C2CN(CN3CSCCSC3)CCO2)=O)CCC(n2cc(CO)nn2)CC1 CC1(C)CCCCCN1C(=O)C(=O)N.N1(CC)CCN(CC(c2ccccc2)O)CC1 c1(NCC2CC(NC(C(CC=C)CC=C)=O)C2)ncnc2onc(C)c12 C1(CC(=O)NCC(CNC(C=C(C)C2CC2)=O)C)CCCS(=O)(=O)C1 N1(C(C(COCC)n2cc(C(N3CCCC3)(C)C)nn2)=O)CCCC(F)CC1 C12C(CC)CCN1C(=O)c1cc(ns1)ONC2=O.c1(OC)cc(COC)[nH]n1 N1(Cc2c(F)c(Br)cc(OC)c2F)CCC2(CC(C(=O)NCCCCl)=NO2)C1 CCC(C)CC(C)CC(C)C(=O)Nc1c(C)[nH]c2ncccc12 c1(C(C(=O)N2CC(CN(C(=O)C(C)n3cccn3)C)C2)SC)ccccc1 CC1CN(C(C2(N=[N+]=[N-])CC2)=O)CCN1C(c1nc(Cl)sc1Cl)=O C=CC(C)(CC)C(=O)NCC12CCC1CN(C(=O)COc1ccccc1)C2 c1(C(N(CCCC(N2C(COC)COCC2)=O)C)=O)cc(C)c(N)cn1 c1(C(=O)NCC2(C)CCN(C(c3cc(O)cs3)=O)CC2)nccn2ccnc12 C(=O)(CC(C)C(C)(C)C)N.C#CCCCCC(=O)N1CC(C2CCC(C)(C)CC2)(O)C1 c1(C(=O)NC2(CCNC(c3cnccc3Cl)=O)CC2)ccc(O)c([N+](=O)[O-])c1 c1(-n2cc(C3N(C(Cc4[nH]cc(C)n4)=O)CCOC3)nn2)ccc2oncc2c1 C1(C2CCN(C(=O)NCC(CCC)OCC)C2)OCC2CCCCC12 Cc1cccc(C(=O)NCc2occc2C(=O)NCC2(O)CCOCC2)n1 C1(C(=O)NCc2cnc(C)s2)CC(C(F)(F)F)CCN1C(=O)CCc1cccs1 CC1(C(=O)NCC(=O)NCC2(CCc3ccc(O)cc3)CCCC2)CNC(=O)C1 C(CCCC(=O)N(CCCNC(C1CCNC(=O)C1)=O)C)SC c1(CC(=O)N(C)CC2(NC(CCOCCN(C)C)=O)CC2)cccnc1Cl N1(C(c2nc(COC)oc2)=O)CC2CC1C2CNC(=O)CCF C(C(N=[N+]=[N-])C(=O)NC(C1CCN(C(C)C(=O)NC(C)(C)CC)CC1)C)OCC c1(C(=O)NC(C=C)CO)ccc(CNC(c2coc(CC)n2)=O)nc1 c1(OC)cccc(N2CCCC(CN(C)C(C3CCCC3C)=O)C2)c1[N+](=O)[O-] C#CC(C)CN=C(NCC(C)(C)C)NC1CCCCC1 CC1OCCN(Cc2ccc(-c3c(F)ccc(O)c3F)cc2)C1(C)C C12CCCCCCN1C2=O.C1(CC(=O)NC(C2(CC)CC2)C)CCSC1 C1(CNC(C2(c3ccc(C)s3)CC2)=O)C2CCCC2CN1C(=O)CCC1(C)N=N1 C(=O)(C1=NN(CCO)C(=O)CC1)NCC(CC)(C)NC(=O)Cc1c(C)noc1Cl C(=O)(C1=NOC2(CCC2)C1)NC1CCC(NC(c2c(C)nc(C#N)cc2)=O)CC1 C1(C(N(C2CCN(C(=O)Cc3cncn3C)C2)CCC)=O)(C(C)C)CCCO1 c1(C(=O)NCC(CN(C(C2C(C=C)C2)=O)C)(C)C)c(NC(C)=O)sc(C)c1C Cc1cc(CN2CCCC2CNC(=O)COCC(F)F)n[nH]1 C1(NC(C(OC)OC)=O)CN(C(c2ccc(OC(F)(F)Cl)cc2)=O)CCC1CO C1(CCN(C(=O)COC(=O)CC)C)CCN(C(C2CC2CCl)=O)CC1.C(C(F)(F)F)O c1(C(=O)NCC2(C)C(NC(Cn3nnc(C)n3)=O)CCC2)nsc2ccccc12 Cc1cccnc1C(=O)NCCC(C)(C)CNC(c1oc(C(F)(F)F)nc1C)=O c1(OC)cnnc(C(N2CCC2C(=O)NCCC2CCC(C)(C)O2)=O)c1 CC(CCNC(=O)C(C)(O)C1CCC1)N=c1[nH]c(Cl)ncc1C#N c1(CNC(C2CCCCC2)C(C)C)ccc2c(c1)CCC2(C)C CCC(CCC(=O)N(CCCC(O)CO)C)NC(c1cn(C)c(=O)cn1)=O C(CC1=CCN(C(C2CC(F)C(=O)N2)=O)CC1)NC(=O)CC1CCCCO1 N1(C(c2n(C(C)C)ncc2)=O)CCN(C(=O)CN2CCC(O)CC2)CC1C(F)F c1(C(N(CCN(C(=O)CC2CCCCC2C)CC)CC)=O)nnn(C)c1C C1(C(N)=O)COCCN(C(C2CCC(C(C)C)N2C(=O)CCCCC2CC2)=O)C1 c1(C(C)=O)cc(Cl)ccc1-c1cn(CC(=O)NC2(C)CCN(C)C2=O)nn1 N1(C(c2cc(SNCC)ncc2)=O)CCC(C)(NC(=O)CCC2(C)CC2)CC1 CC1(C)CN(C(=O)CCc2ccccc2F)CC(CNC(=O)CC2CC23CC3)O1 Cc1cccc(C(=O)NCc2cc(F)ccc2Br)c1O.C12CN(CC1(F)F)C2=O C(=O)(C(F)C(C)CNC(=O)C(C)COC)NCCCOCCC c1(C(N(CCCN(C(C(CC)F)=O)C)C)=O)ccc(OC(C)=O)c(-n2cnnn2)c1 c1(CC(N2C(CNC(C3CN(CC(C)C)C3)=O)COCC2)=O)cccc(C#N)c1 C(C(O)C(=O)N1CC(O)(CC)C1)NC(C1(C#C)CC1)=O C1(C(N)=O)CN(C(=O)CC2CNC(=O)O2)CCC1NC(c1cc(Cl)cnc1O)=O CC1(C)CC(CNC(=O)Cc2ccc(F)cc2F)N(C(C2CCCC2)=O)C1 C1(CC(=O)N(C)Cc2cscn2)N(C(c2ccnn2CCF)=O)CCC1(C)C N1(CC2(C)CCC2)C(=O)CCN(Cc2cccc(-c3ccccc3)c2)C1=O C1(NC(C2CCN(C)C(=O)C2)C)CCN2CCC1(C)C2 CCCCC(CNC(c1c[nH]c(C#N)c1)=O)NC(c1cnc(S)n1C)=O C1(NC(C2C(OCC)CC2)=O)C2CCCN(C(=O)CCP(C)(C)=O)C2C1(C)C c1(OC)ccc(-c2ccc(O)c(C)c2)cc1CNC1CCCN1C(=O)C1CC1 C1(CC(=O)NC)COCCN1CC(=O)Nc1csc(-c2ccccc2)n1 CN=c1[nH]ncn1CC(=O)Nc1ncn(Cc2cccc(F)c2)n1 C(C(=O)NCC#CC(F)(F)F)(C(C)(C)C)NC(c1nc(C)n(C)c1)=O C1(N(C(Cc2c(C)cco2)=O)C)CN(c2ncc(O)cn2)CCC1O C1(C(=O)NC)CN(C(=O)CCCOC(C)(C)C)CCO1.C1(OCC)CC1C(=O)OC c1(-c2ccc(C(=O)NCCC3(NC(C(COC)O)=O)CCC3)[nH]2)ccccc1F N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(NC(c2cc(N)ccc2Cl)=O)C(C)(C)C1 C1(O)(CNC(C(C)Cc2ccccc2Cl)=O)CCCN(C(C2OCCCO2)=O)C1 C1(CN(C(CC)=O)C2CC2)CCN(C(=O)C(C)N(C)C(c2cccs2)=O)CC1 c1(C(N2CCC(O)(CNC(C3CC(C)(C)C3)=O)C2)=O)c(Cl)ccc(F)c1F Cc1ccc(O)c(CC(=O)N(CCC(C)(C)NC(=O)Cc2ccon2)C)c1 CCCCC(C(=O)NCCCCCCF)NC(=O)CCCCNC(C)=O C(=O)(C(C(C)C)Nc1cccnc1)NCCN(C(=O)CC1CCCOCC1)CC Cc1nn(-c2ccc(F)cc2)c(C)c1S(=O)(=O)NC(CO)CC(C)(C)C C1(CC(=O)NC(C#C)(C)C)CCC(C)(C)O1.C(=O)C(C)NC CC(C)C(C)C(=O)NC(CNC(=O)C(C)OC1COC1)C1CCC1 c1(OC)cc(NC(=O)C(c2ccc(Cl)s2)Sc2cccc(Cl)c2)ccc1C#N C1(CNC(c2n(CC)ncc2Cl)=O)CCC(C)CN1C(c1ocnc1C)=O CC(=O)C(C)CC(C)C(=O)N1CCCCC2(CCC2)C1 c1(COCC)ccc(N)c(C(=O)NC2(C(C(=O)NC34CC(C)(C3)C4)C)CC2)c1.OC N1(C(CC(CCC)C)=O)CC(NC(=O)COCC2CC2)CC2(CCOCC2)C1 c1(NC(c2nnnn2CC2CC2)(C)CC2C=CCC2)ccc2c(c1)CCO2 C(=O)(C(N)=O)NCC(C)N(C(COCCOCC)=O)CC C(=O)(C1c2c[nH]nc2CN1C(c1cc2n(n1)CCC2)=O)NCC(C1CCCC1)C c1(NC(c2cnn(-c3ccccc3)c2)=O)nccnc1C(=O)O.C12CC1NC2=O Cc1nn(C)c(C)c1CC(=O)NC1(CNC(=O)CC2CCCC(=O)C2)CCCC1 c1(C(=O)NC(CC)CNC(=O)CC2CCCCO2)n[nH]c(C)c1C c1(OCC(=O)NC(C(C)NC(Cc2scc(C)c2)=O)CO)cccc(Cl)c1C Cc1cccn2nc(C(=O)NC3CN(C(=O)C(C)(C)C)CCC3C)cc12 c1(C(N2CC(CC(=O)OC)C(C)C2)C(=O)NC2(C)CC2)sc(C)c(C)c1C c1(C(=O)NC(C)CCNC(=O)CCN2CCC2)c(F)ccc(Cl)c1F c1(C(N2C(C(N3CCC(C)(CO)C3)=O)CCCC2)=O)ccc(F)c(O)c1 c1(C(=O)NC(CSCC)C(=O)NC23COC(COC)(C2)C3)cncc(C#N)c1 c1(OC)ccc(N(CCOC)CCC2CC2)cc1.C(=O)(N(CCO)C)NC.C1CC1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC(F)(CNC(c2c(OC)ccnc2O)=O)C1 C(=O)(C(C(C)C)NC(=O)C(C)SC(C)(C)C)NCC(=C)Br c1(CC)nccnc1C(=O)NCC(CCOC)NC(=O)C(COC)OC Cc1cc(C)n(C(C)C(N2CCCC(CCNC(=O)CCc3cncs3)C2)=O)n1 N1(C(c2c(C)cc[nH]2)=O)CCC2CCC(NC(=O)CC3CN4CCC3CC4)C1C2 CC1(C)C(NC(=O)CC2(CNC(C3(C)CC=CC3)=O)CC2)CC1(F)F c1(C(=O)O)cc(Cl)c(O)c(S(=O)(=O)NC2(CSc3ccc(O)c(O)c3)CC2)c1 C(=O)(C1=C(C)CCCC1)N1CC(OCC)(CNC(c2cncc(Br)c2C)=O)C1 CC(C)CC(C(=O)NC1(C(=O)NOCCN(C)C)CCN(C)C1)N(C)C N1(C(=O)CCC2CCC2)CCC(C2CCCCN2C(c2nncs2)=O)CC1 CC1(C)CC(CC(N2CCC(CF)(NC(=O)CNC(N)=O)C2)=O)C(=O)O1 CC1=NNC(=O)C1CC(=O)N(C1CN(C(=O)Cc2cccc(O)c2)C1)C C1(C(=O)NCC2(C)OCCN(C(C3CC(O)(CC)C3)=O)C2)CCc2nnnn2C1 Cc1nc(C(N2CC3CC3(CNC(C3(C#N)CC(C)C3)=O)C2)=O)n(C)n1 c1(NC(C)=O)cc(C)c(S(=O)(=O)N2CCCC2(C)C(C)O)c(C)c1 C(=O)(C(C)(C)CCC#N)NC(C)CC1CN(C(C2(O)CCOCC2)=O)C1 C=C1CC(C)(C(=O)NCCN(C2CCCC2)C(=O)COC2CCCC2)C1 c1(OC)ccc(CN2CCCC(C)(C(N3CCN(CCCO)CC3)=O)C2)cc1Br Cc1ccn2cc(C(=O)NC3(CNC(=O)C=Cc4cnc[nH]4)CCC3)nc2c1 c1(Sc2n(C)ccn2)ccc(C(=O)NCC(=O)OCCC2CCC(C)(C)C2)cc1 N1(c2n(CC(C)C3CC3)c(-c3cc(Cl)ncc3F)nn2)CC(=O)N2CCCC2C1 c1(CC)ccccc1C(=O)N(C1CCC(NC(c2cn(C)cc2C)=O)CC1)C C(CN=c1ccn2nccc2[nH]1)(N(C(Cc1c(OC)ccc(F)c1)=O)C)C1CC1 C#CCC(C)C(=O)N1CCCCC1CCNC(=O)CC(c1cccs1)NC(N)=O C1(NC(C(C)=CC)=O)CCCCC1NC(=O)C=CC1CCCN1C C(=O)(C(C)N(C(=O)C=CC(=O)NCCO)C1CC1)NC(COC)C N1(C(c2cnc(NC(C)=O)o2)=O)CCCC(NC(c2cc(C(F)(F)F)on2)=O)C1 n1(CC)c(CCNC(c2ccncc2)CC2CCCCC2)nc2ccccc12 c1(CCC(=O)Nc2cccc(C(=O)Nc3c(C)ncn3C)c2)c(F)cccc1F C1(F)(C(=O)NCc2c(C(N(C(CO)CO)CC)=O)cco2)CC=CCC1 c1(OCC(=O)NCC2CN(C(C3C(C#N)C3)=O)C2)cc(F)ccc1Br N(C1CN(C(=O)C(F)C(C)C)Cc2ccccc21)C(C1CCN(C(C)=O)C1)=O c1(C(N2CCN(C)CC2CNC(C23CC(O)C2C3)=O)=O)c[nH]c2ccc(F)cc12 C1(C(N(c2ccc(O)nc2)C)=O)CC2CC(C1)CN(C(=O)OC(C)(C)C)C2 CP(C)(=O)CN1CC(C(=O)NCCC2(NC(=O)CCC3CC3)CCC2)C1 N1(C(C(CCCC#C)C)=O)CCCC12CCCN(C(=O)C(C)OC(C)(C)C)C2 N1(C(c2c(CCCC)ocn2)=O)CCC(C)N(C(=O)C(C)NS(=O)(=O)CC)CC1 c1(C(=O)NC(C(C(C)C)NC(CCC)=O)C)sc2ncccc2c1Cl N1(C(C(C)(C)OCCOCC)=O)CCCC1C(=O)NC(C)C.C1(C)C(=O)N1 C1(NC(C(CCCC)O)=O)CS(=O)(=O)C2CN(C(=O)C3=CCOCC3)CC12 c1(C(C(=O)NCc2cc(CC)on2)NC(=O)C=C2CCC2)c(C)cccc1Br c1(C(=O)NCC2CCN2C(c2n[nH]c(C3CC3)n2)=O)cc2n(n1)CCCC2O c1(C(N2CC3CC2CN3C(C2SC3C=CC2CC3)=O)=O)c(F)cccc1Cl c1(C(N(C)CCNC(=O)CCCS(N)(=O)=O)=O)cc([N+](=O)[O-])cc2c1OCCO2 Cc1c(F)ccc2[nH]c(C(=O)NC3CCN(C(=O)Cc4ccns4)C34CC4)cc12 CCCCC(O)C(C)C(=O)NC1(CC(=O)NC2CCC3(CC2)N=N3)CCCCC1 Cc1c(C(=O)NCC2CCN(C(=O)CC3CCCC(=O)C3)C2)cnn1CC(C)C N1(C(CCCSC)=O)CCC(NC(c2cc(Cl)nnc2O)=O)C(C)C1 Cc1ccc(C(F)(F)F)cc1C(=O)NC1CC(C(=O)NCCOC(F)(F)F)C1 c1(C(CC(=O)NC(C)CCCNC(C2CCSCC2)=O)C)ccc(N)cc1 CCCCCCC(C)C(=O)NCC(CC)NC(C1CC2C(C1)C2(F)F)=O C(=O)(C(C)(O)C(C)(O)C(=O)NC(c1nc(C(F)(F)F)cs1)C)OCC C1(NC(c2c(C)ccs2)=O)CC=C(C(=O)NCC2CCCSC2)C1 C12CCN(CC1C)C2=O.C(C)(C)(CN(C)C(c1cnsc1)=O)N(C)CC CC1(C)CCN(C(=O)Cc2cnc[nH]2)CC1CNC(c1cn2ccccc2n1)=O C(c1cc2ccccc2o1)=CC(=O)NC1CCN(C(=O)Cc2nnc(O)s2)C1 C1(C#N)(C(N2CC3C(CC(=O)NCCCC=C)C3C2)=O)CCOCC1 C1(NC(=O)CCC2CCC2)CC1C1CCCN(C(c2cnnc(Cl)c2)=O)C1 N1(C(c2cncc(C#C)c2)=O)CCOC2(CCN(C(=O)CCC=C)C2)C1 C1(C(=O)NCCNC(c2cc(C)cc(C)c2N)=O)Cc2cncn2C(=O)N1 C1(C(=O)NCCN(C(C(C)(C)OCC)=O)C)CNC(=O)CC12CCOC2 c1(C(=O)NCC(C)NC(C(C(CC)C)O)=O)ccc2nc[nH]c2n1 N1(C(C2(C=C)CCC2)=O)CC2CC(C1)N(C(c1ccc(C#N)[nH]1)=O)C2 CC1CC(CCNC(=O)CCC2CCOC2)CCN1C(c1cc[nH]c1)=O C(=O)(C1CCc2nnc(C)n21)NCC(C)NC(C1=C(CC)OCCC1)=O C1(NC(CN2CC(C)C2)=O)C=CCN(C(c2ccnc(C(C)(C)C)n2)=O)C1 CC1CN2CCN1C(C(N1CC(CCNC(=O)C(O)CC3CCCC3)C1)=O)C2 CC(C)(CF)C(=O)NC(CNC(c1ccc(-c2ccc(Cl)cc2)[nH]1)=O)C(C)(C)C C1(CC(=O)N(CCCCNC(=O)CCCc2ccccn2)C)CC(C)(C)CCO1 N1(C(CC2CC(OC)C2)=O)CC2CCC(N(C)C(c3ccnn3C3CC3)=O)C2C1 c1(CC)cn2c(n1)CC(C(N1CCC(NC(c3ccc(Br)o3)=O)C(F)C1)=O)CC2 N1(C(=O)OC(C)(C)C)CCCC(F)(CSC2CCCCN2C(c2ccco2)=O)C1 c1(NC(=O)CC2(Nc3ncc(Br)c(O)n3)CCC2)cc(F)cc2[nH]ccc12 C(CN=c1ccnc(NC(c2nc(CC3CC3)n[nH]2)C)[nH]1)C1OCC(C)C1 N1(C(CSC)=O)CCC(CN(C(=O)C(c2ccccc2F)(C)OC)C2CC2)CC1 c1(C(=O)NCCN(C(CN(C(=O)OC)C)=O)C)cnn(C2CCOCC2)c1 C(CN=c1[nH]c(=NCCc2ccc(F)c(F)c2)[nH]c2c1CC(C)CC2)c1c(C)cco1 O=C1CN(CC(=O)NCC23CC(NC(c4nccnc4N)=O)(CO2)C3)C(=O)N1 N1(C(c2ncccc2O)C(=O)NCCC2(C)CC2)CCNC(=O)C1CCN(C)C C=CCC(CC=C)C(=O)NC1(C2CCN(C(=O)C(C)CC(F)(F)F)C2)CC1 c1(OC)ccnc(C(=O)NC2CCN(C(=O)CC3CCC(C)C3)CC2)c1N Cc1[nH]c(=N)nc(O)c1NCC1(c2ccccc2)CN(C)C1 Cc1nc(NC2CCC(NC(c3cnn(CCC(F)(F)F)c3)=O)CC2)[nH]c(=N)n1 C1(O)(C(C(=O)N(C(C)CO)C)NC(=O)CP(C)(C)=O)CCCCC1 CC(C)C(CNC(C12CCC(C1)C2(C)C)=O)C(=O)NCc1nc(O)cc(O)n1 C(=O)(CC(C)(C)C(F)(F)F)N1C(CNC(C2(C)CCNC2=O)=O)CC2(CCC2)C1 c1(CCC)ccc(-c2noc(N3CC(OC)C(OC)C3)n2)cc1 CCCCCC(=O)NC(CNC(=O)CNC(=O)NC)C1CCC1 c1(C(CCC)NC(=O)C(=O)NCCN(C(C)C)C2CC2)cccc(Cl)c1 c1(C(N(C2CN(C(c3ccc(Cl)cc3N)=O)CC2F)C)=O)[nH]cc2c1CCC2 O=[N+]([O-])c1cccc(F)c1CS(=O)(=O)N(c1nccc(N2CCCC2)n1)C1CCNC1 C=CCCC(N=c1cc(C)[nH]c(=NCC(COC)OC)[nH]1)c1ccccc1 C1(C(N(CCNC(C2N(C(=O)OC)CCC2)=O)C(C)C)=O)CNC(=O)C(C)(C)C1 c1(OC)ccnc(CNC2C=CCCCC2)c1 C1(CCC(=O)NCC(F)(F)CO)CCC(NC(=O)CCc2ccco2)CC1 CC(C)C(C)(O)C(=O)NCCC(C)CCNC(c1ccc(C2CCCC2)cc1)=O N1(c2cc(C)ncn2)CCCC(C)(CNC(C2CCCN2C2CCCC2)=O)C1 CC1(C)CC(C(=O)NOCCO)CN(C(C2CC(F)(F)C2)=O)C1 N1(C(CCc2cc(C)no2)=O)CC=C(CNC(C2CCS(=O)(=O)C2)=O)CC1 CC1CCC(C2CC2)N(C(=O)Cc2cocn2)C1 N1(C(C2CN(C)C2)=O)CCC(F)C(NC(=O)C=Cc2ccccc2Br)C1 c1(C(=O)NC2CN(C(C3CCC(C)NC3=O)=O)C2)cnn(C)c1S(N)(=O)=O N1(C(C(C)N(C)C)=O)CCOC2CN(C(c3cnn(C)c3N)=O)CC12 N1(C(C=CC)=O)CCCC2C1CCCCN2C(c1coc(C(C)(C)C)n1)=O C(C)(CN=c1ncnc2n(C)[nH]c(Br)c1-2)NCc1ccc(NC(C)=O)o1 C1(NC(c2ccc(Cl)cc2F)=O)CCC2CC1CN2C(c1n[nH]c2c1CCC2)=O c1(C(=O)NC2CC3(CC(CNC(CC(C)SC)=O)C3)C2)c(F)c(F)cc(F)c1F CCC(CCC(=O)NC)OC(C1CCCN1C(c1cc(C)ccc1F)=O)=O C12(CNC(c3c(C)nns3)=O)CCC1CCN2C(=O)CCCc1ccsc1 N1(C(C(n2cnc(C#N)n2)C)=O)CCC(C)(CNC(=O)C(c2ccccc2)F)C1 c1(C(=O)NCC2(O)CN(C(=O)Cc3ccno3)C2)coc2c(F)c(Cl)ccc12 c1(C(=O)NCC(C)NC(C(c2cnn(C)c2)OC)=O)oncc1C c1(C(=O)NCC(CNC(COCCOCCOC)=O)O)cc(O)ccc1C c1(CC)ccccc1OCC(=O)NC(C1CN(C(=O)Cc2nccn2C)C1)C C1(C(N(CC(CN(C(c2c(C)cc(F)s2)=O)C)O)C)=O)CC2(C1)CC21CCC1 C(=O)(CCCC(=O)NCC1CCCC(NC(=O)CCOC(C)C)C1)OCC Cc1ccc(CNC(C2(NC(C3CCCN3C=O)=O)CCC2)=O)nc1 C1(CNC(C2(C)ON=C(C)C2)=O)CC2(C1)CN(C(=O)CC1CN3CCC1CC3)C2 N1(C(c2nc(CCCC)sc2)=O)CCC2(CNC(=O)COC3CC3)CCCCC12 C(=O)(C1CCc2cccnc21)NCCCN(C(CCC(=O)NC)=O)C Cc1cc(=NC2CCCc3c(OC(F)F)cccc32)[nH]c(Cl)n1 c1(NC(C(COCC)N=[N+]=[N-])=O)cccc2c1OCCO2 CON(C)CCCNC(C1CCN(C(=O)CCC2CCCCO2)C1)=O c1(C(C(=O)NCC2C(C)(C)OCC2)(F)F)cc(C(F)(F)F)cc(F)c1 C(=O)(C1=NN(C)C(=O)CC1)NC1CN(C(C(COCC)C)=O)CC2(C1)CC2 C1(NC(C(C2CN(C(CCSC)=O)C2)O)=O)CCN(CC(=O)OCC2CC2)C1 S(=O)(=O)(c1cccc2c1OC(C)C2)NCc1c(CC)nco1 S(=O)(=O)(c1ccc(-c2ccon2)c(OC)c1)N1CCC(N(CCOC)C)C1 S(=O)(=O)(c1cnc(NCC2CCCC2O)c(Cl)c1)NCC1(C)CCC1 N1(C(C2CN(C(C(C)c3cc[nH]n3)=O)CC2C)=O)CCC(O)CC(C)C1 c1(CN=C(NC(CC)CC)NC(CO)CCF)cn2ccccc2n1 C(=O)(C1c2ccccc2C2CC1C2)N1CCN(C(CCC=C=C)=O)CC1CF c1(C(=O)Nc2c(C)n(C)nc2)cc2n(n1)CCCN(Cc1ccc(Br)cc1F)C2 Cc1ccc(F)c(CNC(=O)NCC(C)(O)CC(C)(C)C)c1Br c1(C(N(C(C#C)C2CC2)C)=O)c[nH]nc1NC(C1(C(C)C)CCC1)=O N1(C(c2cc(Cl)cnc2O)=O)C2CCC1CC(NC(C1(O)CC3CCC1C3)=O)C2 c1(NC(=O)NCC(C)N(C(=O)C(C)C)CC)cccc(F)c1C#N c1(Cc2c(CNC(C)=O)nco2)nc2cc(C)ccc2s1.c12cc(n[nH]1)NC2=O N1(C(C2(NC(=O)Cn3cccn3)CCN(C)C2)=O)CCN2CCOCC2C1 C(=O)(CC(C(=C)C)OCc1ccccc1)N1CCC(NC(C(C)OCC=C)=O)C1 N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C(C)OCCN(C)C)C(C)C1 Cc1cn(CC(=O)NC2CC(CNC(C3CCCCC3C)=O)C2)nc1C(F)(F)F C1(CC(=O)NC(CNC(CC(CCC)O)=O)C2CCC2)CCC2(CCCC2)CC1 C1(F)(CNC(CC2CCN(C)C2)=O)CCCN(C(=O)C(C)(C)O)CC1 N1(C(C2N(C(CN(CCC)C)=O)CCC=C2)=O)CC(C2=NOC(C)C2)C1 C12(OC)CCC(C1)N(C(=O)C(=O)NC1(Cc3cnn[nH]3)CCCC1)C2 c1(C(=O)NCC(CNC(C(CC)Sc2ccccc2)=O)C)cnn(CC)c1F C1(NC(CCc2c(C)n(C)nc2)=O)CN(C(c2cn[nH]c2)=O)CC12CC2 CC(C)C(O)C(C)C(=O)NCC1(NC(C2(CO)CCCC2)=O)CCCCC1.C(N)=O c1(OC)cccc(C(N2CCC=C(CNC(C3(C)CSC3)=O)C2)=O)c1O c1(NC(C(C2CN(C(C3CCC(N(C)C)C3)=O)C2)O)=O)ccc2nccn2c1 N(C(=NCCCCC1CCCC1)NC1CC1)Cc1cn(C)nc1C(F)F C1(C(N2CC(CC(C(N3CCN(C)CC3CO)=O)F)C2)=O)CN2CCC1(C)CC2 c1(NC(C2C(NS(C(C)C)(=O)=O)C2)=O)cccc2c(Cl)ccnc12 CC1(C)CC(C(N2CCC(CF)(NC(c3occc3Cl)=O)C2)=O)CCO1 c1(CN2CCC(N(C)C(C3CCCCO3)=O)C2)cccc(F)c1F C1(CNC(c2c(N(C)C)cncc2)=O)CC2CCC1N2C(c1scnc1Cl)=O c1(NC2CCCC(C(N3CCC(O)C3)=O)C2)ncnc2ncc(Br)cc12 N1(C(c2ccc([N+](=O)[O-])cc2)C(=O)NCC)CCOC2(CCC(F)(F)CC2)C1 c1(C(=O)NC2CC(NC(C3CC34CCC4)=O)C2)ccc(N2CCCCC2)c(F)c1 [N-]=[N+]=Nc1ccc(C(=O)NCC2CC(F)(F)CN2C(C2CCNC(=O)C2)=O)cc1 c1(C(=O)NCC2C3CN(C(COCCC)=O)C2C3)ccc([N+](=O)[O-])[nH]1 n1(CC)nc(C)cc1C(=O)NC(C(=O)NCC1(C(F)(F)F)CC1)C1CCOC1 CC(O)(CC(=O)N1CCCC2(CC(NC(C3CCSCC3)=O)C2)C1)C(F)(F)F CC(C)C(CN(C)C)C(=O)NC1CCC(NC(=O)Cc2cncn2C)CC1 c1(C(=O)NC(C(C(C)C)NC(c2cnccc2Cl)=O)C)cc(O)c(F)cc1N Cn1c(C(=O)NCC(C2CC2)NC(=O)C(=O)Nc2ncc[nH]2)cc2cc(Cl)ccc12 C(=O)(CC1OCc2ccccc21)N1C2CC(CNC(C=C(C)C(C)C)=O)C1CC2 O=C(C1=Cc2ccccc2C1)N1CCn2c(C3CC3)nnc2C1 C1(CNC(c2ocnc2C(F)F)=O)CN(C(c2cnc[nH]2)=O)CCO1 c1(C(=O)NC(CC2CCCN(C(CSCC=C)=O)C2)C)ccc(C(C)C)c(Cl)c1 c1(CCC(=O)NCCN(CCC)C(C2CCC23CCC3)=O)csc2ccccc12 CC(C)C(C)(C(=O)N1CCC1CNC(=O)CCNC(N)=O)c1ccccc1 c1(NC(C2C3CCN(C(C(C)n4ccnn4)=O)CC32)=O)ccc2c(c1)COC2 N1(C(Cc2ncc(OC)nc2)=O)CCCC(NC(=O)CCC=CC(C)C)CC1C Cc1nc2c(s1)CCCC2C(=O)N1CCC(CCNC(=O)CC2CC=CCC2)C1 CC1(C)CC(NC(C2(n3ccnn3)CC2)=O)CC(C)(C)S1(=O)=O CC1(CNC(c2c[nH]nc2Cl)=O)CC(F)(F)CN1C(C1CCc2c[nH]nc2C1)=O c1(C(=O)NC2CC(NC(C3(C)CC=CCC3)=O)C2)ccc(C(F)(F)F)c(F)c1 c1(NC(c2ccnc(NC3C(C)N(C)CC3)n2)=O)ccnc2ccsc12 C1(NC2(C)CN(C(=O)NC(C3CCN(CC(F)(F)F)C3)C)C2)CCC(F)(F)CC1 C(=O)(C1CCc2cc(F)ccc21)N1CCC(C)C(CNC(c2coc(O)n2)=O)C1 CCCC(C)CC(=O)NCCC1CN(C(c2cncc(O)c2)=O)CCO1 C1(C(=O)NCC2(CC)CCCC2)(CC)CCN(C(=O)CCCn2cccc2)C1 C(=O)(C1=CCCCCC1)N(CCC(C(C)C)NC(C1CCC2(CCC2)CO1)=O)C N1(C(c2c(C)cc(C)o2)=O)CCCC(F)(C(=O)NC(c2nccc(O)n2)C)C1 C#Cc1cnc(NC(C2CC2NCc2ccc(C(F)(F)F)c(F)c2)=O)cn1 N1(C(C)=O)CCCC(N=c2cc[nH]cc2S(=O)(=O)NCC2CC(O)C2)CC1 N1(c2n(CCOCC)c(CC)nn2)CCC(C)CC1C1CCC(C)O1 c1(C(=O)NCC2(O)CCC2)cnn2c1CNCC2 C(C1(C)CCOCC1)=CC(=O)NCC1C(NC(Cc2nc(C)sc2)=O)CCC1 CC1CCN(C(c2cnc(C(N)=O)s2)=O)C(C)C1NC(=O)CC1CSC1 c1(CC(=O)NC(CCNC(C(CC=C)C)=O)C)c(F)c(F)cc(F)c1F Cc1cc(=NC2CCCN(C(=O)Cn3cc(C4CC4)nn3)C2)[nH]c(CO)n1 Cc1cc(=O)c(C(=O)NC2CC3CN(C(=O)CC4=NNC(=O)C4)CC3C2)cn1C C(CC(C(C)C)NC(=O)CCCSC)N.C1(C(=O)NC)(C(=O)N(C)C(C)C)CCC1 N1(C(C2(COC)N(C(CC=CCC)=O)CC=C2)=O)CCCN(C=O)CC1 C(=O)(CCC(=O)NN(C)C)NCC(CN(C(C(C1CCCO1)OC)=O)C)(C)C N1(C(c2c(C)noc2C(C)C)=O)CC2CC(NC(=O)CCC3CC3(F)F)C1C2 CC1=C(C(=O)N2CCOC(CNC(=O)CCC3CCOC3)C2)CC1 C(CC(C)C)(C(=O)NOC(c1ccccc1)C)ONC(c1c(C)cc(N)cn1)=O Cc1cc(C(N2CC(C)(CNCc3nccs3)C2)=O)c(F)cc1Br c1(OCC)cccc(C(=O)NC(C2(O)CN(C(=O)CC(C)C3CCCO3)C2)C)c1 C(C)(CCC(=O)NCC1(O)CCC1)NC(c1ccc(CC)[nH]1)=O CC(C)CC(F)C(=O)N1CCCCC1CCNC(C1CCN(S(C)(=O)=O)CC1)=O C(=O)(CC(C)(C)CC(=O)OC)N(CC)CC1CCCC1F.C12CCCN1C2=O c1(CC)nn(C)cc1C(=O)NCC(C)(O)CNC(c1csc(C(C)OC)n1)=O c1(OCCC)cccc(CC(=O)NCC2(OC)CCN(C(=O)C3CC3)C2)c1 Cc1nc(C)n(CCC(=O)NC(C)C(C)NC(C23CC(C#N)(C2)C3)=O)n1 C[Si](C)(C)c1cccc(-c2noc(-c3cccc(C(F)(F)F)c3F)n2)c1 C(C(CC(=O)NC(c1c(C)noc1C)C)OC)NC(C1(CC#C)CCC1)=O C(C(O)CC(=O)NCC1(N(C)C2CC2)CCC1)OCC.C12(CCN(C)C1)C(=O)N2 c1(C(C)NC(=O)NC(C)Cc2ccco2)cccc(-n2cccn2)c1 Cc1nn(C)c(C)c1C(=O)NC1C2CC1N(C(C1SCCS1)=O)C2 CN(CCCCN1CCCCC1)N1CCC(C(=O)NC(=O)C2CC2)C1 C1(NC(CC2(COC)CC2)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)C1C N1(CC)N=C(C(=O)NC2CCC2CNC(c2nn[nH]c2C(F)(F)F)=O)CCC1=O N1(c2cc(C)nc(N3CCCC(CC#N)C3)n2)CC2(CCC2)CC1C N1(C(COCC)=O)CCCC2CN(C(c3ccc(C(F)(F)F)o3)=O)CCC12 c1(C(=O)NCC2CCC3(C(NC(CSCC)=O)C3)CC2)ccc2c(c1)ncn2C C=C1CC2(C1)CC(C(N1CCC1CC(=O)COC)=O)C2 Cc1cnc2ccc(C(=O)NCCN(C(=O)Cc3cc(Br)cs3)C)cn12 N1(C(C(C(C)C)SC)=O)CCC(C(=O)NC2CCCN(C)C2)=C(F)C1 N1(C(C2(C(=O)NC)CCC2)=O)CCC(C)(C(=O)NC2CC(C(F)(F)F)C2)C1 c1(NC(=O)OC(C)(C)C)cc(CCNC2C=CCC2)cc(C(F)(F)F)c1 C1(C(=O)NC(C2(O)CCN(C(=O)COCC3CC3)CC2)C)CCC2(CCCC2)C1 Cn1cnc2cc(C#N)c(COCC3CN(Cc4ccccc4)C(C)(C)C3)nc12 C(=O)(C1=CCC1)NCCN(C(C1CC(C(C)(C)C)C1)=O)Cc1ccccc1 N1(C(C(CC)(C)CNC(c2cc([N+](=O)[O-])c[nH]2)=O)=O)CC2CC(F)CC2C1 N1(C(C(C(C)C)C2CCC2)=O)CCC12CN(CCO)C2 c1(C(C)C)ccc(F)c(C(=O)NC2C3CCN(C(c4cnsc4)=O)C23)c1 c1(NCc2cc([N+](=O)[O-])c(O)cc2)cc(-c2cscn2)nc2ccccc12 C1(CNC(c2ncc(OC)cn2)=O)(NC(=O)CC(C)C(C)C)CCCCC1C CC(C)CCN=C(NCc1ncccc1Cl)N1CCC(C(C)O)C1 C1(CC(=O)OC)(NC(c2cn(-c3ccnc(CO)c3)nn2)(C)C)CCOCC1 O=C(CC1COCc2ccccc21)NC1CCN(C(=O)Cc2ccns2)CC1O c1(C(=O)NC2C3CCN(C(C(CCC)CCC)=O)C32)cnc2cc(O)nn2c1O C1(CNC(C2CN3CCCN2CC3)=O)CCN(C(c2cscc2Cl)=O)CC1(F)F C1(NC(c2c(C)cc(C)nc2)=O)CN(C(=O)Cc2nc[nH]n2)C2CCCC12 c1(C(N2CCC(OC)(CNC(C34CC(C)C3C4)=O)C2)=O)ccc2c(c1)C(C)CN2 c1(N(C)C)c(C(=O)NCCCNC(=O)C(C)(C)C(N)=O)nnc2ccccc12 C(CC(O)C(=O)NC1(C(=O)NCC23CCC(CO2)C3)CC(F)(F)C1)N(C)C n1(CCC)nc(C)cc1C(=O)N(C(CNC(=O)C(C)O)CC)C C1(CNC(Cc2c(C)n(C)nc2)=O)N(C(=O)Cc2cscn2)CCCC1(C)C C1(CNC(Cn2cc(C(C)=O)nn2)=O)CCCCN(C(c2cncnc2)=O)C1 CC(C)(CCCCNC(=O)Cc1cnsc1)C(=O)NNC(=O)c1ccnnc1O C1(OC)CCC(CNC(=O)C(C2CC=CCC2)NC(=O)CN2CCOC2=O)CC1 C1(O)(NC(C(OCC)OCC)=O)CCN(C(C2CC2c2ccco2)=O)C1 n1(CC(C)CO)nc(-c2ccc(C(N(C)CCN(C)C)=O)cc2)nc1CNC=O C1(CNC(=O)CC2CCCCO2)CCCN(C(=O)Cc2nccs2)C1 C1(C(N2CCC(CN3CCCC3)C2)C(=O)NCc2cccs2)(CCC)CC1(C)C c1(C(=O)NCC(CC)NC(=O)Cc2csc(C)n2)c(C)oc(C)c1C CCC(CO)(C(=O)N1CC(O)(CCNC(C2CC3CC3C2)=O)C1)OC N1(C(C2(COC)CC(=C)C2)=O)CCCC2(CCN(C(C3SCCCS3)=O)C2)C1 c1(C(CC)NC(C2(NC(c3conc3C)=O)CCC2)=O)cccnc1 C(=O)(C(C)(C)S(C)(=O)=O)NC1(CC)CN(C(=O)COC2CC(C)CC(C)C2)C1 Cc1ncc(CCC(=O)NC(C)C(CO)NC(c2cnc(N(C)C)s2)=O)s1 c1(NC2C(CC)CN(C)C2)nc2cc[nH]c2c(=NC2CC(OCCOC)C2)[nH]1 N1(C(c2n(CCC#N)ncc2)=O)CCC(CNC(C2(n3cccn3)CC2)=O)CC1 c1(OCC(C)OC)c[nH]nc1CCCC(=O)NC1CC1c1ccco1.C1CO1.COC n1(CCC(=O)NCC2C(NC(CN(C)CC)=O)C2)ncc2c1CCCC2 C=CCCCC(C)(c1nnnn1C(C)CC)Nc1ccc(OC)c(CC)c1 N1(C(c2c(C)cnnc2)=O)C2CCCC1CN(C(c1coc3ccccc13)=O)C2 N1(C(C2CCN(C(C(CC)O)=O)CC2)=O)CCc2c(C#N)cccc21 C1(C(=O)NCC(O)CC2CCCCC2)CCCN(C(=O)Cn2cc(Cl)cn2)C1 C(CCCCCC(=O)NCC1CN(C(C)=O)C1)n1cc(CN(CC=C)CC=C)nn1 C1(NC(C2CCCN(CC)C2)=O)CCN(C(=O)CC2CCCC2)CC1(C)C C1(O)(C(C)NC(c2nocc2Cl)=O)CCN(C(C2COCCOC2)=O)C1 Oc1ccc(-c2ccccc2)cc1CNCc1nnnn1C1CC2CCC1C2 C1(CNC(C(CC)(C)C)=O)CCN(C(C2CCCNS2(=O)=O)=O)C1(C)C Cc1cc(=NCc2cccc(Br)c2F)[nH]c(=NC(CCO)C(F)F)[nH]1 C1(NC(c2ccc(O)cc2)=O)CN(C(=O)C#CC2CCCCO2)CCC12CCC2 c1(NC(C(CCSC)NC(C(CC=CCC)C)=O)=O)ccc(F)c(O)c1 c1(OCC#N)cc(Cl)ccc1CSc1nnc(-c2ccccc2F)s1 c1(SC)cccc(C(=O)NC2CCCCC2NC(=O)Cc2cnnn2C)c1Cl C1(C(N(CCC(=O)N(C(C)C)CC)C)=O)CCC1C(N)=O.C1(=O)C=CCO1 c1(SC)cc(C(=O)NC2CC2CNC(c2ccc(C(N)=O)s2)=O)c(C)o1 c1(C(=O)NCC2C(NC(C(COC)OC)=O)COC2)cccc(CS(N)(=O)=O)c1 c1(OC)ccc(C(=O)C(=O)N(C(c2ccc(O)cc2)CO)C)cc1 C1(CCNC(COCCC)=O)CCN(C(c2coc(Br)n2)=O)C(C)C1 C12(C(=O)NC3C(CNC(Cn4c(C)ncc4)=O)CCC3)CCC(C1)OC2 c1(C(=O)NCC2(O)CC(CNC(CSC)=O)C2)ccn(C)c1C c1(C(=O)NC2(COC)CN(C(=O)CC3CC3C(F)(F)F)C2)c[nH]c(=N)nc1C c1(C(C)OCC)nc(C)c(C(=O)N(CCCCCNC(C2CCOC2C)=O)C)s1 c1(C(=O)NC2CC(CNC(C3(F)CC3)=O)C2)nc2n(c1Cl)CCCC2 N1(C(CCc2cnc(C)s2)=O)CCN(C(c2ccc(CO)nc2)=O)CC1C1CC1 C1(C(=O)NC2(C)CCN(C(C(C)=C(CC)C)=O)CC2)CCN(S(=O)(=O)N(C)C)C1 O=C(C1=C(Cl)CCCC1)NCC1CCC(NC(=O)C(F)(F)C2(O)CCCC2)CC1 C1(CNC(C(COC)C)=O)CCCCC1NC(c1ccn(CC2CC2)c1C)=O C12(NC(C(C)OC)=O)CCOCC1CN(C(c1ccc(Br)cc1F)=O)C2 C1(NC(CC(=O)OC)=O)CC2CCC1N(C(=O)C(CO)C(C)C)C2 c1(C(=O)OCc2nc(C)on2)cc(Cl)ccc1N(C(C)C)Cc1ccccn1 c1(C(=O)NCCCN(C(C2CCCCC2(C)C)=O)CC)nccc2ccccc12 c1(C2N(CC(COc3ccc(OC)cc3)O)CCC2)ncc(F)cc1F C1(CC(N)=O)CCCN(C(=O)C(Cn2cccn2)NC(C2CCOCC2)=O)C1 c1(CN2CC=C(C(=O)Nc3ccc(CO)cc3)C2)ccc2ncnn2c1 c1(OCC(=O)NCC(CC)NC(C2COC(=O)N2C)=O)ccc(C)cc1C C(=O)(C1=Cc2cc(F)ccc2OC1)NCC1CCN(C(CC(C)O)=O)C12CC2 C1(CC)CN(C(C2CN3CCC2CC3)=O)CCN1C(C1CC(CC2CC2)C1)=O C1(CC)COC(C)CN1C(c1ccc(Br)cc1)C(=O)Nc1ccc(F)cc1C N1(CCC(N2CCC(N(C(CC3ON=C(CC)C3)=O)C)C2)=O)CCP(C)(=O)CC1 C1(CNC(c2cnn(CC)n2)=O)CCC(C)CN1C(c1cc(CO)ccn1)=O C1(C(=O)NC(CNC(c2ccc(C#N)o2)=O)CO)CCC2(CCC2)OC1 c1(OC)cccc2cc(C(=O)NCCN(C(=O)CC(C)C(N)=O)C(C)C)c(=O)oc12 C#CCC(CC)NC(=O)C(c1ccoc1)NC(=O)CCOCC(F)F c1(C(O)NC(=O)C2CC2)ccccc1.C1(CNC(=O)OC(C)(C)C)(CO)CCC1 C1(CCCCNC(COCCC=C)=O)CCCN(C(=O)C(F)(F)CO)C1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)C(C)C2)ccccc1P(C)(C)=O N1(C(=O)CCSc2ccc(Br)cc2)CC2(CCCC2)C1C(=O)O N1(C(CC2(C=C)CC2)=O)CC(CN(C(=O)COc2cn[nH]c2)C)C2(CC2)C1 c1(C(N2CCCC(NC(c3ccc(Br)c(F)c3F)C)C2)=O)ccc([N+](=O)[O-])cc1 Cc1ccn(C(C)C(=O)NC(CO)C(=O)NCC2(CO)CC=CC2)n1 C(=O)(CC(C)(C)C(F)F)NC(C(C)C)CCN(C)C(C1CC(C)(C)C1)=O c1(C(=O)NC2(COC)CCN(C(C3CCC3C(C)(C)C)=O)C2)cncn(C)c1=O C1(CC)(CC)CC(NC(c2c(C)csc2Cl)=O)CN1C(=O)CC1CCOC1 CCCCC(CNC(=O)CN1CCCS1(=O)=O)NC(C1CC(C)(C(C)(C)C)C1)=O c1(OCC)cc(Br)ccc1NC(C1CCC(NC(=O)C=Cc2cnccn2)C1)=O N1(C(c2cccc(CC)c2O)=O)CCCN(C(=O)CC(=O)NC2CC2)C(CO)C1 c1(C(N(C)CC2N(C(c3ncc(CC)cn3)=O)CCC2)=O)ccc(Br)cc1O N1(C(CCNC(=O)NC)=O)CC(F)(F)CC1CNC(=O)COC1CC1 C12(C(=O)NC3CC(N(C)C(c4ncn5c4CCC5)=O)C3)CCC(C)(CC1)CO2 CCS(=O)(=O)c1ccc(Cl)cc1C(=O)NCC1CN(C)CCN1C(C1CC1F)=O c1(C(N(CCCNC(=O)CCC2CCC(C)O2)CC)=O)cncc(C(F)F)c1 CCCS(=O)(=O)C(C)C(=O)N(CCN(C(=O)C(C)=C1CCC1)C)C(C)C C1(C(C)NC(C2CC2COC)=O)CCN(C(c2cccc(F)c2)=O)CC1 c1(CN=c2ccc(N3CCC(C(C)C)C3)n[nH]2)c(F)ccc2[nH]cnc12 C(=O)(C(CC(C)CC)NC(=O)CC=CC)N1CC(CC#C)OCC1 CC1CCCC=C1C(=O)NC(C)C(CO)NC(=O)Cc1ccc(F)cc1Br Cc1cc(N)cnc1C(=O)N(C1CCN(C(C2CCC3C2C3(F)F)=O)CC1)C N1(C(C(C)N2CCC2)=O)CC(C)(C)C1C(F)(F)F Cc1cc(C(=O)NCC2(CN(C(=O)C(F)C3CCCC3)C)CC2)c(C)n1C Cc1ccc(C(=O)NCC2C3CCC(C3)N2C(c2n[nH]c(C)c2F)=O)c(C)n1 S(=O)(=O)(c1cnc(N2CCOCC2)nc1)N(C1C(C)N(C)CCC1)CCC#N C1(F)(C(N(CCN(C)C(c2coc(Cn3cccn3)c2)=O)C)=O)CCCOC1 c1(C(=O)NC2CC(C)(CNC(CSC)=O)C2)ccc2c(n1)CCC(C)C2 CC(CC(=O)NC1(C)CC1)C(C)(C)NC(=O)C(O)CC(N)=O c1(C(=O)NCC23CCC2CCN3C(c2ccncn2)=O)cc2c(cn1)OCCO2 N1(C(CC(=C)C)=O)CC(C)OC2(CCN(c3cccc(F)c3C#N)C2)C1 CN1CCN(C(C2CCC2CNC(C23CCN(CC2)C3)=O)=O)CC(O)C1 C1(C(=O)NCC(CCNC(C(CC)N(C)C)=O)OC)CC2(CCC2)CO1 C(=O)(C1=CCC(C)CC1)N(C1CCCN(C(=O)CN2CCOCC2)C1)CC N1(C(CNC(c2c(CC=C)cccc2)=O)=O)CCC2CCCCC2C1 N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(c2ccc(N)c(O)c2)=O)CC12CCCC2 c1(C(=O)NCC(C)NC(c2ccc3ccsc3c2)=O)cnn2c1CC(C)CC2 c1noc(CCC(=O)NC2(CNC(=O)CC3CCC(O)C3)CC2)n1.CC(C)C C1(C(=O)NCC(CNC(=O)CC2CCC2)C(F)(F)F)(NC(C)=O)CCC(C)CC1 C(C(N=[N+]=[N-])C(=O)NC(CC)CC(=O)NCC1CC2CCC(C1)C2)OCC N1(C(C)C2CC2)CC(C(N2CCOCC2CCNC(c2cscn2)=O)=O)CC1=O C(CCCCC(=O)N1CCCC1(C)CNC(c1cc2sccc2[nH]1)=O)OC C1(OCC)COCCC1c1nc[nH]n1.C(=O)(CCCSC)NCC1N(C(C)=O)CC1 C1(CNC(C2(C#N)CC2)=O)CN(C(C2CCN2C2CCCC2)=O)C2(CCC2)C1 CCN(OC)C(=O)CNC(C12CC(CO)(CN1C(c1cc(C#N)cs1)=O)C2)=O C1(NC(COCCCOC)=O)CCC(NC(=O)CN2CCCC2CO)CC1 Cc1[nH]nc(Cl)c1C(c1nnnn1CCOC)NCC1(C)CC=CCC1 N1(C(Cc2c(C)ccs2)=O)CCCC2(CC(NC(c3cn(C)nn3)=O)CO2)C1 N1(C(C2C(C)C2)=O)CCC(NC(=O)Cc2ccc(Cl)cc2C#N)C(F)(F)CC1 O=C(CC(C(F)(F)F)c1ccon1)NCCC1CCN(C(c2ccsn2)=O)C1 N1(C(Cc2ccn(C)n2)=O)CCC2(CCCCC2NC(C2CC2F)=O)C1 c1(CSC)cccnc1C(=O)NC(C)CCN(C)C(c1ncccc1N)=O CC(=O)C(C)CC(C)C(=O)NCC=CC(=O)NCC12CCC(CC1O)C2 CCCCC(CC)C(=O)N(c1ccc(N(C)C)cc1)CCc1ccccn1 c1(NC(CSC(C)=O)=O)cnc(Cl)cc1C(N1C2CCC1COC2)=O C1(N(C(=O)Cc2cccs2)C)CCCC(NC(=O)CC2CCC(C)(C)O2)C1 c1(N2CC(COC)N(C(C3CCCCO3)=O)CC2)ncc2ccccc2n1 Cc1cc(CC(=O)N(CC(C)(C)NC(=O)OC(C)(C)C)C)nc(O)n1 C(=O)(C1=NOC(C)C1)NCC1N(C(c2[nH]cc(C(C)=O)c2)=O)CCC1 N1(C(c2cnc(SC)s2)=O)CC2CCC1C(CNC(=O)CC1CCOC1)C2 c1(CN(C(C)CSc2ccccc2)C(C)Cc2cccs2)cccc(F)c1 c1(C(N2C3(CNC(c4cccnc4)=O)CCC3CC2)=O)coc2ccccc12 c1(N(C)CC2COCC2O)nc2cccc(F)c2c(=NCC2CCCOCC2)[nH]1 N1(C(C(=O)NCC2(C(F)(F)F)CCCC2)=O)CCOC2CCCCC12 c12ccccc1NC2=O.c1(SCCCC)sccc1NC(C1(C(N)=O)CC1)=O N1(C(C2C(C)=CCS2)=O)C2CCC1CN(C(=O)CC1=CCCC1)CC2 C(=O)(C(C)(C1CCC1)NC(c1coc(CO)c1)=O)NCC(C1CCCC1)C C1(c2nnnn2C)(C(=O)NCCc2scc(C)c2)CN(C)CC1C C1(NC(c2c(CC)c[nH]n2)=O)CC2CCC1CN2C(c1cccnc1)=O CS(=O)(=O)C1CN(C(=O)Cn2ncnn2)CC1NC(C1(CO)CC1)=O c1(CN2CC(N(C(c3cc(C)cc(Cl)c3)=O)C)C2)cc([N+](=O)[O-])cc(Br)c1O Cc1cccc(F)c1C(=O)NC1(C(N2CCCC(CC(N)=O)C2)=O)CC1C C(N1CCC(C)(C#N)CC1)N1C(C)CCC(C)(C)C1 c1(C(=O)NCC2(C#N)CN(C(c3ccc(C)n3C)=O)C2)cc2ccccc2[nH]1 C(=O)(C(C(C)(C)C)n1ccnn1)N1CC(C(C)NC(c2csc(O)n2)=O)OCC1 Fc1cccc(CCCC2CCOC2)c1 c1(C(=O)NCC2N(C(CCOC)=O)CC2)cc2cc(F)ccc2[nH]1 C(C(CO)CC(C)C)NC(CN(CC(C)C)C(=O)CC1CCCC(=O)C1)=O N1(C(c2c(C)nc[nH]2)C(=O)Nc2ccccc2Cl)CCC2CCCC2C1 N1(C(CC2CCN(C(c3cnn(C)c3N)=O)CC2)=O)CC(O)CC12CCCC2 c1(C(=O)NCCNC(CC2C(CC)C2)=O)cc(S(=O)(=O)N2CCC2)c[nH]1 CCC(C)C(O)C(=O)NC(C)CCN(C)C(c1cnn(C)c1C(C)(F)F)=O c1(CC(C)(C2CC2)OC(C(F)OC)=O)cc(Cl)ccc1Cl Cc1cccc2c(O)nc(CNC(COC(C)(C)C)CO)nc12 c1(OC)c(Br)cc(CNC2CCN(C(c3ncc(C)n3C)=O)C2)cc1Br S(=O)(=O)(c1ccc(C(=O)N(C)C(c2cc(C)ccc2C)C)cc1)NCC N1(CCC(N2CCC(NC(=O)C(c3ccc(O)cc3)=O)CC2)=O)CCC(O)CC1 c1(C(N2CCN(C(=O)CSC(F)(F)F)CC2)=O)ccc(C2CC2)c(F)c1.C1CC1 N1(C(c2ccn(CC)n2)=O)CCC(CNC(=O)C(n2cc(C)cn2)C)C(F)(F)C1 N1(C(C(=O)N(C2CCCC2)CC(C)C)=O)CC(CO)C2(CCC2)C1 CC1CN(C(=O)C#CCNC(=O)C(F)CC2CCOC2)CCN1C C1(NC(CSCCC)=O)CCC(CNC(=O)C(O)Cc2cn(C)cn2)CC1 c1(CC(=O)NC2CCCC(NC(C(C)OC)=O)C2)cccc([N+](=O)[O-])c1C C1(C(N2CCC(O)(CN(C(=O)C=Cc3ccoc3)C)C2)=O)CCCCCCC1 c1(C(=O)NC2(CNC(CNS(CC)(=O)=O)=O)CCCC2)cc2ccc(F)cc2[nH]1 C(=O)(CCCCC(C)(C)C)N1CCC(NC(C(CC=C)C(C)C)=O)C12CC2 O=C1CC2(CCC2)C(C(N2CCCC2CCNC(C23CCC(CC2)C3)=O)=O)CN1 C1(NC(=O)Cc2cccc(Br)c2)CC2C1CCN2C(=O)CN1CCNC(=O)C1 CCC(F)(F)C(C)(C)C(=O)N(CCC(C(C)C)NC(=O)CCC(C)C)C C1(NC(CC2ON=C(C)C2)=O)CC2(CCC(NC(=O)CCCCC(C)C)CC2)C1 c1(CC)ccc(CCNC(=O)Nc2ncc(-c3cccs3)s2)s1 c1(C(=O)NC2C(NC(C(C)SC)=O)CCC2)ccc2c(c1)N(C)CC2 C1(C(=O)NC2CN(C(c3c(C)scn3)=O)C(C)C2)CC12CCSCC2 N1(c2n(CCC=C)c(-c3cnc4ncccn34)nn2)CCN2CC(C)CC2C1 CC(O)CCN=c1cccc(S(=O)(=O)NCCc2ccncc2)[nH]1 C1(C(=O)NC(CNC(C(CC)Cc2ccc(N)cc2)=O)C)CN(CP(C)(C)=O)C1 Cc1c(C(N2CC3CC(NC(=O)C=Cc4ccccc4)C2C3)=O)sc2nccn12 C(C(CNC(C1CC2(CSC2)C1)=O)S(C)(=O)=O)NC(CCN(CC)CC)=O Cc1c(C(N2CCC(N(C(=O)CSC3CC3)C)C2)=O)[nH]c2c(C)cccc12 C=CC(C)(CC)C(=O)NC(C)CC(C)NC(c1nc(Cl)ccc1Cl)=O CC1Cc2cccc(C(=O)NCC(O)CCNC(=O)CSc3n[nH]c(=N)s3)c2O1 c1(OC)cc(C(N2CCC(NC(=O)C3=CCC3)C(C(C)C)C2)=O)ccc1Cl c1(OCCC(=O)NC2CCC(NC(CC#N)=O)C2)ccccc1F C(=O)(CCCCC(C)CC)NCC(=C)CCNC(c1cc(Cl)cc(Cl)c1)=O C1(NC(C(C)C)=O)CCCC(NC(c2ccccc2-n2ccnn2)=O)C1 C1(C(=O)NC2CC3N(C(C(C)=O)=O)C(CC3)C2)CCC2(CCOCC2)O1 C(=O)(C1=NN2CCCN=C2N1)NCC1(CNC(c2cc(C)n(C)n2)=O)CC1(F)F N1(C(c2c(C)coc2C)=O)CC2=C(C1)CN(C(=O)C(C)c1cncs1)C2 c1(C(=O)NCC2N(C(=O)CC3(C(F)(F)F)CCC3)CC=C2)cc2n(n1)CCCN2 C1(NC(C2(C#C)CCCC2)=O)CC12CCN(C(c1coc(CO)c1)=O)CC2 CC(CC(=O)NCC1C=CC(NC(=O)CNC(C2CCC2)=O)C1)C(C)(C)C C12(CNC(c3c(CC)n(CC)nc3)=O)CC(CO1)N(C(C1CC1CC)=O)C2 CC(C)CC(C)C(=O)N1CCCC1CCNC(=O)CC1(CS(C)(=O)=O)CC1 n1(CC(=O)NC(C)(CNC(c2coc(Br)n2)=O)C2CC2)cnc([N+](=O)[O-])n1 N1(C(c2cccc(C(=O)NC)c2)=O)CC(C)CN(C(c2ncoc2C)=O)CC1C N1(C(C(CC=C)NC(C)=O)=O)CC2(CCCC2)C1C(N1CC2CC2C1)=O CC1=C(C)CC(C(=O)NC(C)(C)C=CC(N2CCC(C(C)(C)C)CC2)=O)CC1 c1(CNC(c2cccc(NC(c3ccnc(O)c3)=O)c2)=O)ccc2csnc2c1 c1(NCC(=O)NCCOCCNC(C2CCC2)=O)csc(-c2ccco2)n1 C(=O)(C1=CCOCC1)NCC1C(C)(C)C(NC(c2cc(-c3ccco3)[nH]n2)=O)C1 c1(OC)ccccc1C(=O)NCCCCCCN(C)C(C1CC(C)(C)O1)=O N1(C(C2N(C(CCc3onc(C)n3)=O)CC2)=O)CCCC(O)C1C C=CC1CN(C(c2c[nH]c(=NCC)s2)=O)CC1NC(=O)C(c1c(C)n[nH]c1C)C c1(C(N2CC(C(C)NC(=O)CCn3cncn3)OCC2)=O)cc(Cl)c2n[nH]cc2c1 N1(C(COc2cn(C)nc2)=O)CC2CCC1C1CN(C(=O)CCC(N)=O)CC21 c1(C(=O)NC(C)C(=O)N(C2CCCCC2C)C)ccccc1Br c1(C(=O)NC2CCCN(C(c3cncnc3)=O)C2)cc2ccc(O)nc2s1 Cc1sc(N)c(C(N2CCC(C)(CNC(c3ccc(O)nc3Cl)=O)C2)=O)c1C C(CNC(C1(C)CC(NC(c2cc(CCO)on2)=O)C1)=O)(C(F)(F)F)OC C1(CCNC(C2C(=C)C2)=O)CSCCN1C(=O)C=C1CCCC1 C(=O)(C(F)(F)C1CC1)NCC(CC)NC(C1CN(C2CCOC2)C1)=O C(CC(C)(C)C)(C(=O)NC1(CN(C)C(c2sc(C)nc2C)=O)CC1)OC c1(CCC)onc(C)c1C(=O)N(CCC(=O)NC(c1ccccc1O)C)C1CC1 N1(C(c2cccc(C)c2Cl)=O)CCC2(CCN(C(=O)CC3CC3C)CC2)C1 c1(C(N)=O)cccc(CN2CCC(C(=O)NCc3ccncc3F)C2)c1 C1(NC(C(CC=C)CC)=O)CN(C(=O)CCc2cccc(O)n2)CCC1(C)C C1(CN(C(C2CN(C(C)C)C2)=O)C)C2CN(C(C3(C)CC3(F)F)=O)CC12 C(=O)(CS(=O)(=O)C1CCCC1)OC(C)(C)C.CC1CC(=O)OCC1(C)C C1(CNC(c2c(C)nccn2)=O)CC2(CCN(C(=O)C(C)(O)CC(C)C)CC2)C1 c1(NC(C(C2(O)CCCCC2)NC(C=C(CCC)C)=O)=O)ccc(N=[N+]=[N-])cc1 c1(OC)cc(SC)ccc1CNCC(O)COC1CCS(=O)(=O)C1 C1(CC)(NC(=O)CC2(CO)CC2)CCCN(C(=O)C=Cc2cccnc2C)C1 c1(C(=O)NC(CN(C(=O)CCCN2C(=O)CCC2=O)CC)C)ccc(Cl)cc1F Cc1cc(C(N2CCN(C(=O)CCC(C)(C)C)CC2)=O)nc2ccccc12 C1(CNC(CC(CCC)C)=O)CCC2CN(C(C3(C#N)CCOC3)=O)CC12 N1(C(c2cnc(CC)[nH]2)=O)CC(NC(C2(C#N)CCCOC2)=O)CC12CCCC2 S(=O)(=O)(c1cnn2ccc(NCC(C)C(F)(F)F)nc12)NC1CC(C)=C(C)CC1 N1(S(C)(=O)=O)CCCC(C(N2CC3CC3(NC(C34COC(CF)(C3)C4)=O)C2)=O)C1 c1(CC)nc2c(C(=O)NCCC(C)NC(=O)C(C)CSC)ccnc2[nH]1 C1(NC(c2ccc(C(OC)OC)o2)=O)CCN(C(=O)CC2(C)OCCO2)CC1 c1(OC)sc(C(=O)NCC(O)CN(C(=O)CC(C)OC)C)cc1Br c1(C(N(CCOC)CCNC(c2cnn[nH]2)=O)=O)ccc(COC)cc1Cl Cc1ccc2c(c1)C(N)C(NC(N1CCN(C(c3ccccc3)=O)CC1)=O)C2 N1(C(c2c(Cl)cc(C)nc2)=O)CC(NC(c2oc(C)nc2C)=O)C(S(C)(=O)=O)C1 c1(C(=O)NC(CNC(c2cnn3ccsc23)=O)CO)c(Cl)ccc(F)c1F c1(CC(=O)NCCC(=C)CNC(=O)Cc2sccc2C)ncccc1C c1(C(=O)NC2C(C)(NC(C3CN(C)C(=O)C3)=O)CCC2)cncn(C)c1=O C(C)(CO)(C(=O)NC1CC(CC2CC2)C1)NC(C(=O)NC(C)C)=O N1(C(C=CSC)=O)CCN(CC(C)NC(C2CN(CC(F)(F)F)C2)=O)CC1 N1(C(C2CC(C#C)(O)C2)=O)CC2(CC(NC(=O)C(C)OCCOC)CO2)C1 C1(C(=O)NC(CSCC)C(=O)NCC2(C)CCN(C)C2)CCCN(C)C1 C1(OC)CN(C(=O)CN2CCCCCC2)CC1NC(=O)CC1CCSC1 N(C(=NCC1CC(C(C)(C)C)C1)N1CCC2(C)C(C1)C2(Cl)Cl)C(C)C N1(C(COCCC)=O)CCN(C(c2csnn2)=O)C(c2nccn2C)C1 c1(OC)c(OC)cc(NC(c2cnc(C)c(C#N)c2)=O)cc1SC c1(-n2c(C(C)CCO)nc(CCCC)n2)ccc(C(F)(F)F)cc1Cl CC1CN(C(c2cscn2)=O)CCC1NC(=O)C(c1ccccc1Cl)(F)F C1(C)(CCNC(C=C2CCN(C)C2)=O)CCN(C(=O)CCc2ccc(O)cc2)C1 N1(C(C2(C)CC(C)C2)=O)CCC(CCCNC(=O)CC2CCCOC2)CC1 C1(NC(COC)=O)CN(C(=O)C(C)Cc2ccc(Cl)cc2)CC12CCC2 C1(N(C(C(C2CCCCC2)C)=O)CCNC(=O)C(C)(C)F)CCOCC1 Cc1cc(S(=O)(=O)NCCCC(C)C)cc(C(=O)O)c1I c1(C(=O)NCC23C(CN(C(c4nnc(C)s4)=O)C2)C3)c(O)nnc2c1CCC2 Cc1cc(C(=O)NCCC2CC(NC(c3[nH]c(C)nc3C)=O)C2)c(O)nn1 N1(C(c2n(C)nnc2)=O)CCC2(CCCN(C(C3CC3C(N)=O)=O)C2)C1 C(=O)(CCCc1ccccc1)N1C(CNC(C2C(CC)C2)=O)CC1 C(=O)(C(CO)NC(=O)CNC1(O)CCSC1)NCC1N(C(C)(C)C)CC1 c1(OCC)ncc(C(=O)NC2CCCC(C(=O)NCCSC)C2)cn1 c1(CC(=O)NC(C)CNC(=O)CNC(c2cccc(F)c2)=O)cccc(Br)c1 CC#CC1CCN(C(=O)CC2CC2CNC(c2c[nH]cc2C(C)C)=O)CC1 c1(C(N2CCCC(O)(CC(=O)OC)C2)=O)cc(C)nc2[nH]nc(C)c12 c1(CC)nc(C(N2CCC(NC(C3CN(CC)CCO3)=O)CC2)=O)c(N)s1 c1(CCC(=O)NC(C(C)C)CNC(=O)C(C)c2ncco2)ccc(C#N)cc1F c1(CC(=O)NC2(CC3CC34CC4)CC2)cccc(O)c1 CN1CCOCC1CC(=O)NCC1CC(C(F)(F)F)CN1C(=O)CCCC#N N1(C(c2cc(C)sc2N)=O)CCC2CCN(C(C3CN(C)CCO3)=O)CC12 C1(C)(C(C)C)CCN1C(c1ccc(CNC(c2ccccc2)=O)s1)=O c1(C(=O)NC2CCCN(C(c3n[nH]c(C)c3C)=O)CC2)nnn2c1CCCCC2 c1(OC(C)C(=O)NCC(C)(CO)NC(c2ccc(O)cc2)=O)ccc(Cl)c(Cl)c1 N1(C(C2C(C)CN(C(c3ns[nH]c3=O)=O)C2)=O)CC2(CCC2)OCC1C C1(CC(=O)N(CCNC(=O)C(O)c2ccco2)CC)(COC)CCCC1 N1(CCN(S(=O)(=O)CC)CC)CCN(C(c2cnc(O)n2C)=O)CC1C N1(C(c2c(CNC(c3ccc(CC)cc3)=O)ocn2)=O)CCOC(C)C1C CCC(C#N)(CC)C(=O)N1CC(N(C(=O)C=CCO)C)C2(CC2)C1 Cc1ccnc(O)c1C(N1CCC(O)C(N(C(=O)CCOC2CCCC2)C)C1)=O CC(C)(C)CC(C(=O)N1CCCC1CF)NC(c1ccsc1)=O N1(C(C(N2CCC(COC)CC2)=O)=O)CCc2ccccc2C1.C1(C)CN1C N1(C(C(CNC(C(C(C)C)SCC)=O)O)=O)CC2(CC(O)C2)C1 CN1CCCC1C(=O)NC1(CO)CN(C(=O)C(C)(C)Oc2ccccc2)C1 c1(C(=O)NC(C2CCOC2)C#C)cc(CNC(=O)Cc2cnsc2)ccn1 C(=O)(CC(C)(C)C(C)(F)F)NC(C)CCNC(C1(c2ccccc2)CCOC1)=O CCC(O)C(=O)NC(CNC(=O)OC(C)(C)C)CCOC.C(C)(C)(C)O c1(C(=O)NC(C(=O)N(C(CCCC)C)C)C(N)=O)ccnc(C)c1N c1(COC)nc(C(=O)NC(C)(C)CCNC(=O)C(C)CC2CCCC2)cs1 c1(C(=O)NC2CCCN(C(c3c(C)sc(O)n3)=O)C2C)cnn2ccn(C)c12 c1(OC)nn(C)cc1CNC(=O)C(=O)NCC(c1ccncc1)O C(CC(=O)NCC)(NC(COC)=O)OCC(c1cn(NC(C)=O)nn1)O.N(C)(C)C C=CCC(CNC(c1cnnn1C)=O)C(=O)N1CCC(N2CC=CC2)C1 C1(NC(CC=CCC)=O)C2CC1N(C(C1(N(C)Cc3ccccc3)CC1)=O)C2C N1(C(C2(N(C)C)CC2)=O)CCOCC(C)(CNC(C2(CC3CCC3)CC2)=O)C1 C1(C(N2CCC(CN(C)CC)C2)=O)CC2(CCN1C(=O)CN(C)C(N)=O)CC2 CC(C)C(N=c1[nH]c(Cl)nc(C(C)(C)C)c1C(N)=O)C(C)N(C)C C1(CN(C(=O)C(c2ccccc2)NC(C2CC2(Cl)Cl)=O)C)CCCC1(C)C C(=O)(CCS(N)(=O)=O)NC(C(=O)Nc1ccc(OCC)cc1)=O C1(C)(CN(C(c2ccco2)=O)CC)CCN1C(=O)CCn1cc(C)cn1 NC1(CNc2cc(Cc3ccc(F)cc3Cl)ncn2)CCCS(=O)(=O)C1 C=CCCCC(C)NC(C1(CNC(=O)C(CN(C)C)N(C)C)CC(C)(C)C1)=O C(=O)(CCCC(C)(C)C)N(CC(=O)N(C1CCCC1C)C)CCC N1(C(C(C(C)C)SCC)=O)CC(C(F)(F)F)OC(CNC(c2cc(Cl)no2)=O)C1 C=CCN=C(NCC1CNC(=O)O1)NCC1CN(S(=O)(=O)C(F)F)CCO1 c1(-c2cccc(SC)c2)ccc2cc(C(=O)NC34CCN(CC3)C4)sc2c1 C(=O)(CC(F)(F)C(C)C)NC1C(NC(C(C)(C2CC2)OC)=O)CC1 C1(C(=O)NC(CCC)CC)CCN(C(=O)CC2CC(C)=NO2)C(C)C1 c1(OC(C(=O)NCCN(C(C2(OC)CC2)=O)C)C)ccccc1C Cc1ncn(C)c(=O)c1C(=O)NC1CS(=O)(=O)CC1NC(=O)CC(C1CC1)C1CC1 c1(NC(C(c2cc(Br)c(Cl)s2)N(C(C(CC)C)C)C)=O)cccc(OC)c1 c1(CC(=O)NCc2c(CCNC(C)=O)ocn2)cccc2cnccc12 c1(NCCCN(C(C)=O)C)cc(S(=O)(=O)NCC(O)C2CCC2)ccc1C#N C1(COC)(NC(=O)CCF)CCN(C(=O)C(C(C)C)Sc2ccccc2)C1 N1(C(c2ccc(CNC(C(CC#C)C3CC3)=O)s2)=O)C2CCC1CC(F)C2 C(=O)(C(CC)CCOC)NC(C(=O)NCc1c(CC)nn[nH]1)C N(C1CN(C(=O)CC2CCCC(F)(F)C2)Cc2ccccc21)C(C(=O)NCC)=O c1(-c2nc(CCC(=O)Nc3nc(CCC)c(CC)s3)on2)cc(Cl)nc(Cl)c1 CC(C)(C)C(=O)NCC(=O)NCCCNC(=O)C(N1CCCC1)N1CCCC1 c1(N2C(CC)COC(C)C2)[nH]c(=NCC(C)(C)CS(C)(=O)=O)nc2scnc12 N1(C(COCCC)=O)CC(F)CC1CNC(c1noc(CC)c1C)=O c1(CCC(C)=O)cn(C2CN(C(C3CCCC3OC(F)F)=O)C2)nn1 c1(C2C(C(=O)NCCNC(C3(C)CCCO3)=O)C2)ccc(Br)nc1 N1(C(C23C(C)OC(C)(C2)C3)=O)CCCC12CCN(C(=O)CN(C)C)C2 N1(C(C(c2cccc(C)c2)O)=O)CCC(NC(C2CCCN2C(N)=O)=O)C2CC12 C1(C2CCCO2)(C(N2CC(NC(c3cnc(Cl)s3)=O)CC3(C2)CC3)=O)CCCO1 CC(CCN(C)C)C(=O)NCC1CN(c2ncns2)CCO1 c1(OC)ccc(C(=O)NCC(CNC(C23CCC(CO2)C3)=O)CO)cn1 Cc1cccc2cc(C(N3CCC(C)N(c4nccc(CO)n4)CC3)=O)oc12 C(=O)(CS(C)(=O)=O)NCC(C(=O)NC(C)Cn1ccnc1)N(C)C N1(C(CC2(OC)CC2)=O)C2CCC1CC(F)(CNC(=O)CCCCC(C)(C)C)C2 N1(CCCCNC(C(F)=C(C)C)=O)CCCN(C(=O)CN2CC=CC2)CC1 C1(CCNC(C2CC(O)(CNC(CCc3n(C)cnn3)=O)C2)=O)CCCC2CC12 CN1N=C(C(=O)NC2CC3CC(C2)N(C(c2ccc(NC=O)cc2)=O)C3)CCC1=O N1(CC)CCC(C(=O)NCC2(NC(=O)CC#N)CC2)C1 N1(C(C2N(C(C(C)C(C)(C)C)=O)CCCC2)=O)C2CCC1CC(CO)C2 C(N=c1ccn(CC(=O)NCCCF)c(O)n1)c1ccc(OC)c(C)c1C N1(C(c2ccccc2S)=O)CCC2(CCN(Cc3cccc(Cl)c3)C2)C1 c1(C(C(=O)N(CC(C)NC(c2ncccc2O)=O)C)=O)cc(O)nc(O)n1 c1(C(=O)OC)ccc(CCNC(C2(CC(F)F)CC2)=O)nc1.N(C=O)CC1CC1 C1(CCNC(C2C(C(C)(C)C)C2)=O)CCN(C(=O)CNc2ccccc2)CC1 c1(C(=O)NCC(CN(C(c2c(CC)nns2)=O)C)O)ccc(OC)c([N+](=O)[O-])c1 C1C(N(C)C)C(=O)N1.C(=O)(C(CSC)c1ccccc1)N(CC=C)C N1(C(C2ON=C(C)C2)=O)CC(NC(C2CC(C(F)(F)F)C2)=O)C(C2CC2)C1 N1(C(C(C)n2cncn2)=O)CCN(C(c2nncn2C2CC2)=O)CC1CF C(C1=NOC2(CCC2)C1)NC(C1N(C(C2(CC)CCCO2)=O)CC(=O)C1)=O c12ccc(cn1)-n1cc-2nn1.C1(CNC(C2CCC(OC)C2)=O)C2CCC1CC2 C1(C(=O)Nc2cc(-n3cc(CNC(CC)=O)nn3)ncc2)CCC(F)(F)CC1 Cc1cc(NC(=O)C(=O)NCC2C3(C(=O)OC(C)(C)C)CC(C2)C3)cnc1O c1(NC(N(C)Cc2c(OC)cccc2C)=O)ccc2ncccc2c1 C1(OC)CC(C(N(CCCn2cnnc2C)Cc2cc[nH]n2)=O)N(C(C)(C)C)C1 CC1CN(C(=O)CC(CC2CC2)NC(=O)C(C)(O)C2CC2)CC(=O)N1 c1(C(N(CCNC(=O)CC2COC(=O)C2)CC)=O)ccc2c(c1)OCCO2 C1(CNC(C2CCC(C)CC2)=O)CCN(C(=O)C(c2cccnc2)C)CC1(F)F C1(CN(C(C(C)SCC)=O)C)CCC(NC(=O)CC2CCCC(C3CC3)O2)CC1 CC1C(C(=O)N2CCC(NC(C3COC(=O)O3)=O)CC2)=Cc2ccccc21 c1(NC(c2cc(C)n(C)n2)=O)nc2ccc(N)cc2s1.N12CC3C(C3C1)C2 C(=O)(CCC(=O)NN(C)C)N1CCC(F)(C(=O)NC(C)CCO)C1 c1(C(N2CCN(C(c3c(SC)scc3)=O)CC(O)C2)=O)cccc2ncn(C)c12 c1(C(C)N(C(=O)C(=O)NC(C)C(=O)NC2CC2)C)cccc(O)c1 c1(NC2C(=C)COC2)cc(-n2ccnc2)cc(Cl)c1 C1(C(=O)OC)CCC(C(C)C)N1C(C1(O)CN(C(c2c[nH]c(C#N)c2)=O)C1)=O c1(C(=O)NCCCNC(C2CC2(COC)COC)=O)ccc2c(c1)C1CCC2O1 c1(CN(CCCNC(c2c(C)nns2)=O)C(C)C)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCCCN(C(C2CC=CC2)=O)CC)ccc2c(c1)NC(=O)CS2 c1(CNC(C2C(CNC(C3CCOC3)=O)C2)=O)ccc(-c2cccnc2)cc1 C(c1cc(C)ccn1)=CC(=O)Nc1c(OC)ccnc1 N1(C(CCC(=O)NCC)=O)CC2CCCC(C1)N2C(=O)C(CC)c1ccccc1 c1(CC(=O)NCC(CNC(C(c2ccccc2)NC(N)=O)=O)F)ccc(O)cc1 n1(CC)nccc1C=CC(N1CC(NC(c2cc(C)oc2C)=O)C(O)C1)=O CCCCC(O)C(=O)NC1CCC(C(=O)Nc2cnc[nH]2)C1 c1(C(=O)NC2C(C)N(C(=O)CC3CCOC3)CC2)cc2ccc(F)cc2o1 N1(C(C2CCN(C(=O)NCC)C2)=O)CCCC(C(C)NC(C23CC(CO2)C3)=O)C1 Cc1cc(=NC(=O)CN(C)CC2C3CN(c4cc(Cl)ncn4)CC23)[nH]o1 C1(C(N2CC(CNC(C3CC(C)(F)C3)=O)OCC2)=O)Cc2ccncc2C1 N1(C(CC(C)(C)O)=O)CCCCC(NC(c2ccnc(O)c2)=O)CC1 c1(CC(C)C)ccccc1C(=O)NCCC1CN(C(=O)COC(C)(C)C)CC1F c1(C(C(=O)NCC(N(C(c2c(CC)c[nH]n2)=O)C)C2CC2)O)cccc(C)c1 c1(NC(C2(CC#C)CC=CCC2)=O)ccc2sc(S)nc2c1 C#CC(C)(C)C(=O)NCC1CCC1NC(=O)C(F)C(C)C N1(C(CCCC=C)=O)CCC2CCN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2C1 CC(F)(F)CCC(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)CC(O)C1 C1(NC(c2cnc(OCC)s2)=O)CCCN(C(c2sccc2C#N)=O)C1 CC1CCc2c(C(N3CCCC(N(CCF)C(=O)C4CC4)C3)=O)csc2C1 O=C1CCC(C(=O)N2CC3C(CNC(C45CCCCC(F)(C4)C5)=O)C3C2)=NN1 C=CC1(CC(=O)NC(c2ncnn2C)C)CN(C(c2cnnn2C2CC2)=O)C1 C1(C(=O)NC(CC#C)CC#C)CC(F)(F)CN1C(=O)CCCC(=O)N(C)C c1(CNC(=O)NCCCOCCCN(C)CC)cnoc1CC(C)C C1(N(C(CC2N(CC(C)C)CCC2)=O)C)CN(C(=O)C2CC2)CC1(C)C c1(C(N(C(C)CNC(c2[nH]nnc2C2CC2)=O)C)=O)c(O)ccc(Cl)c1F c1(CN=C(NC(C#C)COC)NC(C)C(=O)OC)ccc2ncccc2c1 N1(C(C2(CC#C)CCC2)=O)CC2CCC1C(CNC(C1CCC(C(N)=O)O1)=O)C2 CCC(C)CC(C(=O)N1CC(C(=O)OC)C1)NC(c1ccncc1F)=O C1(C(=O)NC(CNC(c2nc(C(C)C)sc2)=O)C)CC2(COCCO2)C1 N1(C(c2c(CC)ocn2)=O)CCC(CNC(C2CSC2)=O)C(O)C1 c1(C(=O)OC(C)(C)C)cc(F)c(C(=O)NCc2c(C(=O)OC)cccc2)c(F)c1 c1(C(N2CC(NC(=O)OC)C2)=O)cc(Cl)cc(OC)c1OC.c12ccnc(c1)S2 C1(CNC(=O)CSCCc2ccccc2)CN(C(C2(F)CCOC2)=O)CC1(F)F CN1CC(=O)NC(CC(=O)OCCNC2(c3ccc(Cl)c(N)c3)CC2)C1=O c1(OC)ncccc1CCNC(C1(C(C)NC(=O)C(C)OC(C)=O)CC1)=O Cc1ncc2n1CCN(C(C1COC(CNC(c3cccc4ccoc34)=O)C1)=O)C2 N1(CCNC(=O)OC)CC2CC1CN2C(=O)CCc1cnc(OC(C)C)cn1 c1(C=O)ccc2nncn2c1.C1(CC)CCN(C(=O)CC2COCC2O)CC1 c1(C(N(S(CCN(C)C)(=O)=O)C)=O)nn(-c2ccccc2)c2c1CCCC2 N1(C(CCNC(C(C)(C)C)=O)=O)CC2CC1CN(C(=O)CCN1CCOCC1)C2 CCCC(CC)CCC(=O)N(CCCN(C)C(C1CCC(F)CC1)=O)C N1(C(C(F)=C(C)C)=O)CC(O)(CCNC(c2cnsn2)=O)C1 c1(C(=O)NCC2CCCN2C(c2c[nH]nc2C2CCCCC2)=O)c[nH]ccc1=O c1(NC(C2CN(Cc3cccc(C=C)c3)CC(F)C2)=O)cc(F)cc(C#N)c1 CC(F)(F)C(F)(F)CC(=O)NCC1(C)CN(C(=O)Cc2sc(O)nc2O)CCO1 Cc1cc(=O)c(C(N2CCN(C(=O)CC3(O)CCCCC3)CCC2C)=O)cn1C c1(CC)ccc(Br)cc1NC(=O)OCC(=O)NCc1ccccc1OC N1(C(c2cccnc2)=O)CCC(F)(F)C(C(=O)Nc2ccccn2)C1 c1(OC)cnc(F)c(C(=O)NCC2C3CN(C(C4(C#N)CCSCC4)=O)CC23)c1 N1(C(C=Cc2ccc(CC)cc2)=O)CCCC2(CCN(C(=O)CCSC)C2)C1 C(=O)(C(CC(F)F)c1ccccc1)N(CCCNC(=O)Cc1nc(=N)[nH][nH]1)CC C(=O)(CCCC(=O)N1CC(CNC(c2conc2C2CCC2)=O)C2CC12)NCC CC1(F)CCCCN(C(=NCc2ccnc(-n3cncn3)c2)NC2CC2)C1 c1(C(N(CCNC(C(C)OCC)=O)CC)=O)ccc(F)c2ccccc12 c1(C(N2CCC(NC(CC=C)=O)(CF)C2)=O)cc(C)nc(C)c1 C1(CNC(c2cc(CC)[nH]n2)=O)CCCCN(C(c2nncn2CC)=O)C1 C1(OC)CC(CNC(=O)CCCn2ccnc2)N(C(=O)CCN2CCOCC2)C1 C1(NC(c2c(C)nc(CC3CC3)o2)=O)CC2CC(NC(=O)C(C)CN(C)C)C2C1 n1(CC)nc(C(C)C)cc1C(=O)NC(C)C(C)NC(=O)Cn1cccnc1=O CCCC(CCC)C(=O)NCC1(OC)CN(C(=O)Cn2c(C)cc(O)cc2=O)C1 C(CC(C(=O)Nc1ccc(Cl)cc1)NC(=O)CC1(C#N)CC1)=CC N1(C(c2cccc(SCC#C)c2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C(C)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)CC2CC3(CC3)C2)ccc([N+](=O)[O-])[nH]1 c1(OC)cc2cc3[nH]c2cc1CC(CC)CCC1n2c-3nc(n2)C(C)C1(F)F c1(OC)cccc(C)c1C(N1CC(C(C)NC(c2csc(Cl)c2)=O)C1)=O C1(CC)CN(C(C2CC2(C)C)=O)CCC1NC(=O)CN(CCCCCC)C C1(CC)CCN(C(=O)C(O)CC2CCCC2)C1C(=O)NCC1(O)CCN(C)C1 Cc1cccc(C)c1C(=O)N(CCCCCNC(C12CCCC1CC2)=O)C(C)C C1(CC(=O)NC2C=CCN(C(c3cc(CSCC)on3)=O)C2)CN2CCC1CC2 N1(C(C=Cc2cncc(C)c2)=O)CC2(COC(CNC(=O)C(O)C3CCC3)C2)C1 C1(NC(C2C(c3n(C)ncc3)C2)=O)CCCN(C(C2CC23CCCC3)=O)CC1 C(C(C)(CC(C)C)NC(=O)C1=NOC(C(C)(C)C)C1)NC(c1c(C)cc(C)s1)=O N1(C(CCC=C)=O)CCN(C(C2CC(=O)N(C(C)CCC)C2)=O)C2(CC2)C1 C#CCC(C)(C(=O)N(CC(C)N(C)C(C)=O)C)NC(=O)CC(COC)COC c1(NC(=O)NC(C(CC)C)Cc2ccccc2)cc(C)c(OC(F)F)c(C)c1 C(=O)(N=c1cc[nH]c(C)c1)c1c(C)sc(-c2ccc(OC(F)(F)F)cc2)n1 c1(C(=O)NCC2N(C(C(CC)OC)=O)CC(F)(F)C2)ccc(F)c2ccccc12 N1(C(C(CC2CCC2)NC(C2C(C(C)(C)C)CC2)=O)=O)CCNC(=O)CC1C c1(C(C)NC(C(=O)NC2CCCN(C(CC(C)C)=O)C2)=O)ccc(C#N)c(Cl)c1 N1(C(=O)C(N2CC3CC3C2)=O)CCOCC1C1CCC1.c12nocc1C2 CCC(C)C(C(=O)Nc1nnc(-c2nn[nH]n2)s1)N1CCCC1 C1(NC(CCNC(=O)CO)=O)CN(C(C2CC2C2CC2)=O)C2(CCCC2)C1 C1(NC(c2ccc(C(C)F)cc2)=O)CN(C(=O)CCCC#N)C2(CCCOC2)C1 c1(OC)ccc(Cl)c(C(=O)NCC(C2CCCC2)NC(COC(=O)CO)=O)n1 Cc1cc([N+](=O)[O-])ncc1C(=O)Nc1ccc2c(c1)COC2 C=CC1CCCN(C(c2ccnc(CNC(c3ccsc3C#N)=O)c2)=O)C1 c1(OC)ccc(NC(N2CCCC(n3cnc(C#N)n3)C2)=O)c(OC)c1Br c1(C(=O)Nc2c(F)cc(C(C)=O)c(C)c2)cc(C2=CCSCC2)n[nH]1 c1(C(=O)NCC2C(NC(C3C(C)C3)=O)CCCC2)cc(S(N)(=O)=O)c[nH]1 C1(C2CCCC2)(C(N2CCOC3CN(C(CCCSC)=O)CC32)=O)CCNC1=O N1(C(=O)Nc2c(C)cno2)CCN(C(=O)C(N2CCSCC2)C)CC(C)C1 C(C1CCN(C(C2CC2(C)C(F)F)=O)CC1)=CC(=O)N(C1CC(C)C1)C c1(CNC(c2c(C(C)C)nco2)=O)ccccc1CNC(C1CCCC12CC2)=O C1(NC(c2nc(C)c(C)s2)=O)CC2CN(C(=O)C(C)C3CC3)CC2C1 N1(C(C(COC)OC)=O)CCC2(CCCC2Nc2cc(=O)n3nccc3[nH]2)CC1 C1(CC(N2CC(NC(c3c(NCC)scn3)=O)C(F)C2)=O)CCC2(CC1)CC2 CC1CCC(Cl)=C(C(=O)N(C2CC23CC3)C)C1 c1(C(N2CCC(CNC(CCCCCC)=O)C23CC3)=O)cc(=NC)[nH]cc1Br C1(CC(=O)NCC(C2CC2)NC(Cc2cn(C)nc2)=O)C2CCCCCC12 C1(NC(CC2CC(OC)C2)=O)CN(C(c2ccc(C(C)(C)C)cc2)=O)CCC1C C1(C(N2C(C(N(CCCCO)CC)=O)CCC2)=O)CCCC2CCCCC12 C1(CCC)CCCN1C(=O)CCC1(NC(=O)COC2CCOC2)CCC1 C1(CNC(CC(C)OC)=O)CC(NC(c2ncsc2C2CC2)=O)C(O)C1 C(=O)(C(C(=O)N1CCC(NC(=O)CCCNC(=O)OCC2CC2)CC1)OC)OC Cc1cccc2c1C(NCC(O)C(F)F)CCC2 c1(C(=O)NC(C(C(C)C)NC(C(=Cc2ccco2)C)=O)C)ncn2c1CCCC2 Cc1cccc(F)c1C(=O)NC1(CC(N)=O)CCN(C(=O)C=CC=C(Cl)Cl)CC1 C1(C(=O)NCc2c(OC)nsc2)CC2C=CC1N(C(=O)CC1CCSC1)C2 c1(C(N(C2CCN(Cc3nccc(C)n3)C2)CCC)=O)cc(C(C)=O)oc1C C1(CNC(C(CC)(F)F)=O)CCN(C(c2cccc(C(C)C)c2F)=O)CC1C S(=O)(=O)(c1cc(C(=O)O)cc(Cl)c1)N(C1CCNCC1)C.C1(N)CCNC1(C)C c1(C(=O)NC2CC(C)(NC(C3CC3C(F)F)=O)C2)ccnc(C(F)(F)F)c1 CC1C(NC(c2cc(C(F)(F)F)ccn2)=O)CCCN1C(c1cnsc1)=O CN1CCN(C(c2ocnc2-c2ccccc2)=O)CC1CNC(=O)C(N)=O c1(C(=O)NCCC(C)NC(c2ncnc(O)c2Cl)=O)cccc2c1NCCC2 c1(C(=O)NC2CC(NC(COC)=O)C23CCC3)nnn2cc(C)nc(O)c12 Cn1cncc1CNC(=O)C(Cc1ccco1)NC(=O)CC1CCCSC1 CC1=NOC(C(N2CCC2CNC(c2ccnc(C)c2)=O)=O)C1C CCC(C)C(C(=O)NCc1ccccc1Br)NC(=O)Cc1nccn1C c1(C(N2CCC(O)(CN(C(=O)C=Cc3ccoc3)C)C2)=O)ccsc1S(N)(=O)=O c1(C(=O)NC2(CNC(C3C(C=C)CC3)=O)CC2)ccc(CCOC)nc1O N1(C(C(CCCC)NC(c2ccnn2C)=O)=O)Cc2c[nH]nc2C(C)C1 C1(C(N2CCC(CS(CC=C)(=O)=O)C2)=O)C=CC(=O)N=N1 c1(C(=O)NC2C(NC(C(C(C)C)OCC)=O)CC2)cc2cc(Cl)ccc2n1C C1(C(N(CCCNC(=O)Cc2cscn2)C)=O)CCCN1C1CCCCC1 C(CCC)(CCC)NC(CC1(N(C(CCC=CC)=O)C)CC1)=O c1(C(N2CCC(CS(C)(=O)=O)C2)C(=O)NC)ccn(CC(F)(F)F)n1 C1(OC)CC(CNC(C2(C)CS(=O)(=O)C2)=O)N(C(=O)CCCc2csc(C)n2)C1 C1(O)(CNC(=O)CC(O)C2CC2)CCCN(C(=O)C(F)n2cccn2)C1 CN1CCc2nc(C(=O)NC3CC4CC3N(C(=O)CCc3cn[nH]c3)C4)sc2C1 C(C)(CN=c1ccnc(NC(CC(F)F)c2ccccc2)[nH]1)OC C1(O)(CNC(c2c(CCC)nns2)=O)CCN(C(=O)C(N2CCOC2=O)C)CC1 c1(C(=O)NC2C3CCC(CN(C(C(CC)C)=O)C3)C2)cncc2c(F)cccc12 CC(C)C(O)CC(=O)N1CC2(CO)CC1(C(=O)NCC(c1ccccc1)O)C2 S(=O)(=O)(c1ccc(=NCCS(=O)(=O)NC)[nH]c1)Nc1c(NCCCC)cccc1 CC1CCN(CCn2cc(C3CN(C(=O)CC4CNC(=O)O4)C3)nn2)C1 c1(NCC2C(C)COCC2)ccc(S(=O)(=O)NCC2(CC3CCC3)CC2)c(Br)c1 c1(C(N2CC(CCNC(=O)CCF)(OC)C2)=O)c(Cl)ccc2cc(CO)cnc12 c1(C(=O)NC2C3CC(NC(c4c(C)con4)=O)CC32)cccc2ccn(C)c12 c1(C(C)C)cccc(OC(=O)C(C)N(C)CC2CCS(=O)(=O)C2)c1 c1(C(N2CC(NCc3c(OC)cccc3F)C(C)C2)=O)csc2ccncc12 C(=O)(CCCC(=O)OC)N(C1CCN(C(=O)CNC=O)CC1)CC#C C1(CCNC(Cc2ccc(N)cc2)=O)CN(C(C2(C(N)=O)CC2)=O)CCCO1 CC(C)CC(CNC(=O)C(C)(C)NS(C)(=O)=O)NC(C1(C2CCCCO2)CC1)=O c1(COC)noc(NC(=O)NC(Cc2nccs2)Cc2ccccc2)n1 C1(NC(C2(C)CCSCC2)=O)CCC2(CCN(C(c3cccnn3)=O)C2)C1 c1(C(=O)NCC(C)NC(CC(C)F)=O)cc2c(nn1)CCCO2 CN1CCCC(CC(N2CCC(C(C)(C)C)(CNC(=O)C(C)(C)CF)C2)=O)C1 C1(C(N2CC(C(C(C)C)O)C2)=O)CCCCCN1C(=O)CC1OCCO1 c1(C(=O)NCC(C)(CO)NC(=O)Cc2cscn2)ccc(-c2coc(O)n2)cc1 c1(C(N2CCN(C(c3cc(F)cc(Cl)c3)=O)C(CO)C2)=O)cc(Cl)cnc1Br N1(C(Cn2c(CCC)ncc2)=O)CC2CCC1CN2C(=O)CC1CCCOCC1 C=C(C)CC(C(=O)NCc1cnc(C)s1)NC(=O)C(C)CCCOC Cc1occ(C(F)(F)F)c1CC(=O)N(CCNC(C1CCCOCC1)=O)C(C)C C(CC(C(=O)NCc1ccc(C)nc1)NC(=O)CC1CCCC1O)SC c1(C2C(C(N(CC(C)NC(CSC(C)C)=O)C)=O)C2)cn[nH]c1 C(=O)(C(C)(C)C(O)C(C)C)N1CC(OC)(CNC(=O)C=Cc2cccc(F)c2)C1 C1(NC(C2(CC)CC2)=O)CN(C(c2ccc(N)c(C)c2Cl)=O)Cc2nccn2C1 C1(C)(OC)CCCC1N=c1[nH]c(N2CCCC(NC(C)=O)C2)nc2ccccc12 N#Cc1c(F)cc(C(=O)NC2CCCC2NC(=O)Cc2cccnc2Cl)cc1F N1(C(Cc2c(C)noc2Cl)=O)CC2CCC(C1CO)N2C(c1ccoc1)=O N12CCc3sc(nc3C1)C2=O.c1(NC(C)=O)ccc2c(c1)CCCC2 CN1C(=O)c2ccccc2C1C(=O)N1CC2(NC(C3CC3F)=O)CCC1CC2 C1(C(C)C)(C(=O)N(C(CO)C2(O)CC2)C)CCN(C(C2CN(C(C)C)C2)=O)C1 c1(C(N2CCCC2CCC2CCCN(C(c3cnco3)=O)C2)=O)ncccc1O c1(-c2nc(C3OCCC3)nn2C(C)C(C)(C)C)n[nH]c2c1CC(C)(C)CC2 CCCC(CCCS(C)(=O)=O)C(=O)N1CCN(C(C)(C)C2=CC3CC2C3)CC1 C(c1ccccn1)=C(C(=O)NCC(C)CNC(=O)Cn1cnnc1O)C c1(C(=O)NC(C2CCCC2)CNC(=O)CCN2CCCC2)nccn2cccc12 c1(C(=O)NCC2C3CN(C(C4CC45CC(O)C5)=O)CC23)cn2c(n1)CCCC2 Cc1ccc(-c2ccc(C(=O)N(C)CC3CCCN(C)C3)o2)cn1 C1(c2c(C(=O)NCC(C(C)O)C)c[nH]n2)CCCCN1C(c1cnsc1)=O c1(C(C(=O)NCC(=C)C)N(CC(=O)NCC)CCOC)cc(Cl)ccc1Cl CCCC(C(=O)NC1COCC1C(=O)NC)NC(c1ncccc1CC)=O Cc1cc(C(=O)NCC(C2CC2)NC(c2cnn(CC(F)F)c2)=O)cs1 N1(C(c2snc(C)c2N)=O)CCC2CCN(C(c3coc(O)n3)=O)C2C1 CC12CC(C(N3CC(=C(F)CNC(=O)CCC4CC4(C)C)C3)=O)(C1)C1(COC1)O2 c1(CCC)ccc(NCC(=O)NC23C(C(=O)NC)CC(CC2)C3)c([N+](=O)[O-])c1 n1(CC(N2CC(N(C(C(CC)OC)=O)C)C3(C2)CC3)=O)c(C)nc2ccccc12 c1(NC(C2CC(F)CN2C(c2ccccn2)=O)=O)cc(F)c(Cl)cn1 C(CCCC(C)(C)C(=O)NNC(=O)C1CC1Cl)NC(C1CCCCN(C)C1=O)=O CC(C)(C(=O)N1CC2CC2(NC(C2C3CCC(F)(F)C23)=O)C1)C(N)=O C1(C(=O)NCC(CNC(=O)C=CCO)O)CC12C1CC3CC(C1)CC2C3 n12c(nnc1S)C(C(C)C)NC(=O)CC2.N1(CC)CCCOC1 N1(C(C(COC)C(F)(F)F)=O)CCCC2(CCN(C(=O)CSC(C)C)CC2)C1 C12CCC(C)CN1C(=O)C1CC(O)(C1)CNC2=O.C1(CC)CCCCCN1C CC1OC(C)(C)OC1(C)C(=O)NCC1(F)CN(C(c2ccnnc2O)=O)C1 c1(C(N2CC(NC(c3cc(CC)on3)=O)C(C#N)C2)=O)cnc2cc(Cl)ccn12 C(N=c1ccc(S(=O)(=O)NC2CCC2O)c[nH]1)c1cccc(S(=O)(=O)NC)c1 c1(C(=O)NCC2(F)CN(C(=O)CC3(CO)CC3)C2)c[nH]c2ccncc12 C1(COC)CC(CNC(=O)CCC2(O)CCC2)N(C(=O)CCCn2cccn2)C1 c1(CCN2CCN(S(CC(=O)OC(C)(C)C)(=O)=O)CC2)cc2ccccc2o1 c1(C(=O)OCC)cc2c(C)nn(CC)c2s1.c1(NCC=O)ccc(CN(C)C)cc1 c1(C(=O)OC)no[nH]c1=NC(=O)C1(F)CCN(C(c2cnc(Br)s2)=O)CC1 c1(NC(=O)Nc2c(C(=O)OC)cc(Br)cc2C)cc(C)c(F)cc1Br N1(C(c2c(C(C)C)occ2)=O)CCC2CCN(C(C3CC(F)(CO)C3)=O)CC2C1 C1(NC(C=CSC)=O)CN(C(=O)CC2CCCCO2)CC1c1ccc(F)cc1 CCCC(C(=O)NC(CCN(C)C)C(=O)N1CCC(CCN(C)C)C1)NC(C)=O C1(N(C(c2n(CCC)nc(C)c2)=O)C)CC2CCC(C1)N2C(c1cc(Cl)c[nH]1)=O c1(C(=O)NCC(C(CC)CC)N2CCCC2)cc2ccc(F)cc2nc1O N1(C(CC)=O)CCCC2(CCN(C(C3(C)COC(C)CO3)=O)C2)C1 c1(C(=O)NC(C(C)C)CCN(C)C(c2cnccn2)=O)cc2c(F)cccc2[nH]1 O(NC(=O)N=c1[nH]nc(SC)s1)CCc1c(CC)cccc1 CC12CCCCC1CN2C(=O)CC(O)COCOC.C(=O)(CSC(F)F)NC1CC1 C(=O)(C(CC(C)(C)C)OCC)N(CCOC)CCNC(=O)Cc1ccc(C)nc1 c1(C(=O)NCC(C2CCN(C(C3CCC3)=O)CC2)(C)C)ccc(Br)cc1N Cc1cccc2c(C(=O)NC3CC3NC(=O)CSCC3CCCCO3)n[nH]c12 CC1(NC(c2cc[nH]n2)=O)CCCN(C(C2CCCS2(=O)=O)=O)C1 Cc1cccc2c1OCCC2Nc1ccc(NC(C)C2CC2)nc1 c1(C(=O)NCCC2(C(N(C3CCCC3)CC#C)=O)CCCC2)cnc(S)nc1 c1(C(c2nnnn2C2COC2)NCc2n(CC)cnc2)ccccc1Br C1(NC(c2ccc(=N)[nH]c2)=O)CC2(C1)CN(C(C1(O)CC1)=O)C2 N1(C(C2(NC(C3N(CC)CC3)=O)CC(O)C2)=O)CC2CN(C)CC2C1 CC1CN(C)CC1C(N1CCCCC1CCNC(=O)C=CC1CCCC1)=O C1(C)(C(N2CC(NC(c3c(C)cc(F)cc3)=O)C(C)(C)C2)=O)CCC(C)C1(C)C N1(C(COC)=O)CC(CNC(C2(Br)CC2(F)F)=O)(OC)C1 CCCCC(CC)CC(=O)NCCCC(C)(C)C(=O)NCC#CC1CC1 CC(C(C)C(=O)N(CCC(F)(F)F)C)NC(c1cccc(=O)o1)=O C1(F)(CNC(=O)CC2CCOC2)CCN(C(=O)CSCc2cccs2)C1 c1(OC)cc(F)c(C(=O)NC2COCCN(C(=O)CCNS(C)(=O)=O)C2)c(F)c1 c1(CC(=O)NCC2(F)COCCN(C(=O)C3=COCC3)C2)ccc2sccc2c1 n1(Cc2snc(COC)n2)c(N2CCC(OCc3cccc(F)c3)C2)nnc1C c1(C(=O)NCCn2cc(-c3ccc(C)cc3)nn2)coc2c1CS(=O)(=O)C2 C(=O)(C1=CC2(CCOCC2)C1)NCC1N(C(C2CC(=C)C2)=O)CCC(C)(C)C1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCC2CN(C(c3n[nH]c(=N)s3)=O)CC12 c1(CN(C(c2nccc(OC)c2)=O)C2CC2)cc2ccccc2o1 c1(C(N2CC(NC(C3CC(CC)OCC3)=O)C(C)(C)C2)=O)ccc(S(C)(=O)=O)o1 c1(NC(CC)CSC)ncnc2cc(Br)c([N+](=O)[O-])cc12 C(CNC(=O)Cc1sccc1C)(C(C)(C)C)NC(COCCOCC#C)=O C(=O)(N=c1ccn(CC2CC2)[nH]1)C1CCCC(NC(C(CCC)F)=O)CC1 N1(C(CN(CC)CCOC(C)(C)C)=O)CCCC2CN(C(=O)C(C)=C3CC3)CCC12 c1(C(=O)NC(C(=O)NCc2c(CC)noc2)C(C)OC)nn(C)cc1C N1(C(CC(CCC)C)=O)CC2=C(C1)CN(C(=O)CCCCNC(N)=O)C2 CCC(CC(=O)Nc1nnnn1C)O.c1(C(N(C)CC2CC2)=O)cc(CO)[nH]n1 C(=O)(C(C(F)(F)F)OC(c1ccccc1)=O)NCC(C)N(C)C C1(OC)CC(C(N2CCN(CCCCCNC(=O)CC3CC3)CC2)=O)CC1OC C(C(F)(F)C(=O)NCC(C)N(C)C(c1cccc(CC(=O)OC)c1)=O)OC CCCCC(C(=O)NC1CC(CNC(c2cc(F)cc(F)c2)=O)C1)N(C)C C1(C2CCN(C(c3conc3C3CCCN3C3CC3)=O)C2)(NC(=O)C=C(Cl)Cl)CC1 C1(C(=O)NC2CC(C)(NC(CCCC)=O)C2)CNC(=O)CC1C C12CCN(CC1)C(=O)CC(C)O2.c1(C(=O)NC2C(C(=O)OC)CC2)cc(C)co1 CN1CC(=O)NCC1C(N1CCOCC1CNC(=O)C(c1ccc(F)cc1)F)=O c1(C(=O)NCCCc2cn(Cc3cccc(C)n3)nn2)ccc2ncn(C)c2c1 C1(NC(c2nnnn2CC(F)F)(C)Cc2ccco2)C2CCCC1CC2 CCC(CC(C)CO)Nc1ncnc(NC2CC(N3CCCC3)C2)c1C c1(OCC(=O)NC(N2CCC(SC)C2)=O)ccc(F)cc1.C1(=O)C(C)OCCN1 C1(CNC(c2c(C)n[nH]c2)=O)CN(C(c2cc(C3CC3)on2)=O)CCCO1 C(C)(C(C(=O)NC1CC(O)C1)C(C)C)NC(c1n(CCC)ncc1)=O c1(C(N(CCOC)CCNC(c2n[nH]cc2C)=O)=O)oc(CC(C)C)nc1C C1(NC(c2c(C)coc2)=O)C2CC3CN(C(c4cn(CC(N)=O)nn4)=O)C1C3C2 Cc1cccc(F)c1C(N1CCC(N(C(=O)CCc2cc[nH]n2)C)CC1)=O C1(NC(C(CC)CC(F)F)=O)CCC2(CC1)CN(C(c1csnc1C)=O)CCO2 n1(CC(=O)NC(CC)CN(C(=O)C(C2CCCC2)OC)CC)nc(C)c(Cl)c1C C1(C(=O)NC(CCC)CO)C2CCC(C2)C1NC(c1nc(C)oc1C)=O C#CCC(C(=O)NCCC1(NC(c2cc(C3CC3)ccn2)=O)CC1)C1CC1 C1(C(=O)OC)CC(c2nnnn2CC(F)F)(Nc2cnc(CSC)nc2)CCC1 C1(CNC(Cc2c(C)n(C)nc2)=O)CC2(CCN(C(c3cnns3)=O)C2)CO1 C1(CC)(NC(=O)CCCCn2ccnn2)CCN(CC2(n3cccn3)CC2)CC1 C1(O)(C(C)NC(C(C)SC(F)(F)F)=O)CCN(C(=O)CCCF)C1 N1(C(C(COC)COC)=O)C(C)CC2CN(C(=O)CSc3ccc(Cl)cc3)CC12 c1(CC(=O)NC2CN(C(C3CC3CF)=O)C3(CCC3)C2)c[nH]c2cccc(F)c12 C1(CNC(C2(COC)CC2)=O)CC2(C1)CN(C(=O)Cc1cncc(Cl)n1)C2 Cc1nc(C(=O)NC(C2(O)CCN(C(=O)Cc3ccn(C)n3)C2)C)sc1C N1(C(c2cn(CC(C)C)nn2)CNS(CC)(=O)=O)CCS(=O)(=O)CC1 c1(C(=O)NCC(C)CNC(C2(Cl)CC2(C)C)=O)ccc([N+](=O)[O-])c(O)c1 n1(CC)nc(C)cc1C(=O)N(CC(=O)NCCc1nc[nH]n1)C1CC1 c1(NC(C2C(NC(C=CC(C)C)=O)CCC2)=O)cccc([N+](=O)[O-])c1F CN(C)NC(=O)CCC(=O)NC(CC1CC1)C(N1CCC(N=[N+]=[N-])C1)=O c1(OC)cncc(CCC(=O)NCC2CCCCC2NC(C2C3COCC23)=O)c1 N1(C(C(C2CCN(C(C3C4CCC(F)C34)=O)C2)C)=O)CCC2CCC(C1)S2 C1(O)(CCNC(C(c2cnn(C)c2)C)=O)CCCN(C(=O)CN(C)C(=O)OC)C1 Cn1cc(C#N)cc1C(=O)N(CC(=O)NCC(O)C(C)(C)C)C1CC1 C(N=c1[nH]c(C)nc(Cl)c1C)C1OCCCN(C(c2c(CCC)n[nH]c2)=O)C1 CCCC(CCC)C(=O)N1CCCC(NC(c2cnc3[nH]cncc2-3)=O)C1 c1(C(=O)NCC2C(NC(c3cc4c(s3)CCC4)=O)C2)cccc(C(F)F)c1Cl CC1CN(C(=O)CC2=CCOCC2)CC(C)C1NC(c1snc(Cl)c1Cl)=O C(CC)(CCCC(=O)NCC(C)N(C)CC)NC(C(C)OCCC=C)=O C1(C(=O)OC)C(F)(F)C12CC(C(=O)NCCC(C)(C)NC(c1coc(C)n1)=O)C2 C1(NC(CC=C=C)=O)CC(CNC(C2(CCN3CCCCC3)CC2)=O)C1(C)C C1(c2cc(CNC(C(C)O)=O)on2)CCN(C(c2cc[n+]([O-])cc2)=O)CC1 C(c1ccc(=N)[nH]c1)=CC(=O)NC(C)CC(C)NC(=O)C(N1CCCC(O)C1)C C1(O)(C(C)NC(C(CCC)N(C)C)=O)CCN(C(c2ccsc2Cl)=O)CC1 N1(C(C(c2ccc(F)cc2)OC)=O)CCOC(CN(C)C(c2ccnnc2)=O)C1 C(=O)(C(C)(C)CN1C(COC)CC1)NCCN(CC)CC.O(C)CC.OC c1(CNC2CC(C(N(C)CC3(C#N)CC3)=O)C2)sccc1Cl C1(C(=O)N(C)CCc2cscn2)(NC(C=CSC)=O)CCSC1 C1(C2CCCN(C(=O)COC3CC=CC3)C2)(NC(=O)Cc2cnoc2)CC1 Cc1cnc(NC2CCN(C(=O)CC3COCCO3)CC2)nc1 CC1CN(C(C2COCC2NC(C2C3CCC(F)(F)C23)=O)=O)CC(C)(C)C1 C1(NC(C(C(C)C)S)=O)CCOC2(CCN(C(=O)CC3CCC3)CC2)C1 c1(N(C2CC3CC2CN3)C(C)=O)cc(S(=O)(=O)NC2CC2(C)C)ccc1Cl c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(C#N)s2)=O)ccc(F)cc1 C1(C(=O)Nc2cc(SC)ncc2)CCC2CCC1N2C(c1[nH]ccc(=O)c1C)=O c1(C(N2C(CNC(C3(C)CC(=C)C3)=O)CC2)=O)cnc(-n2cccn2)cn1 Cc1nn(CC(=O)NC(C)C(C)NC(c2ccc(F)c(O)c2)=O)cc1[N+](=O)[O-] Cc1cc(Cl)c(C(=O)NCCCOC2CCN(C(C3CCCO3)=O)CC2)cc1N N1(C(=O)C=CCN2CCOCC2)CC2CCN(C(C3CCCCC3O)=O)C2C1 C1(C(=O)N(C2(CC)CC2)C)(CC)CN(C=O)C1.C1(=O)CO1.C(C(F)F)O C(C(=O)N(C)CC1CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1)(C(C)C)OC N1(C(C2CCC(C(=O)OC)C2)=O)CCC(C2CN(C(=O)C=CBr)C2)CC1 C1(CC(=O)N(C2CCN(C(=O)CCCCC3CC3)CC2)C)CCCCC12CC2 c1(C(=O)NCC23CC2CN(C(c2ncc(Cl)cc2Cl)=O)C3)c[nH]c2ncccc12 N1(C(C2(C(=O)NC)CC2)=O)CCC2(CCN(C(C34COC(OC)(C3)C4)=O)C2)C1 CC1CN(C(c2ccccc2Cl)=O)CC1CCNC(c1cnc(N(C)C)o1)=O C(CC(C)C(F)(F)F)SC1OCC(C(=O)N(CCC=O)CCO)C1.CO CCCC(C)(CCC)C(=O)NC1CC2C(NC(c3ccc(C(C)=O)cc3)=O)C2C1 c1(C(=O)OC)ccc(C(=O)N(C)CC2CCCN2C(C2(CC(C)C)CC2)=O)o1 N1(C(C2(C)CSC2)=O)CCCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1 CC(C)C(C)C(CNC(C1CC12CCCC2)=O)NC(=O)Cc1cc(F)ccc1F CC(CC(=O)NC1CCCN(C(c2cc(-c3ccncc3)n[nH]2)=O)C1)C(C)(C)C C(=O)(CCCCc1cnc[nH]1)N1CCC(C2(NC(C3C(C)C3(F)F)=O)CC2)C1 C1(C(N2CC(C(N3CC4(CC(O)C4)C3)=O)C(F)(F)C2)=O)CC2C(C1)C2(C)C C(=O)(C(CC(F)F)N(C)CCC1CCCC1)C(=O)CC1CCOCC1.C(COC)N N1(C(CCCC#CC)=O)CC2CC(C(N3CCC(O)C3(C)C)=O)C(C2)C1 N1(C(C(=O)NCCNC(C(C)C)=O)=O)CCCC([Si](C)(C)C)C1 c1(C(=O)OCC)cc(Cl)c(NC(=O)CN2CCC(F)(F)C(C(N)=O)C2)c(Cl)c1 C(=O)(CC(F)(F)Br)NC(CNC(C(CC)c1ccccc1)=O)(C)CO c1(OC)ccc(C(N2CC(CNC(c3nncn3C)=O)C(C)C2)=O)cc1 C=C1CC(C)(C(=O)NC2CC(NC(=O)C(O)Cc3[nH]cnc3C)C2)C1 C1(CC)CCOC1CNC(=O)OC(C)(C)C.C12CCN(C1)CC(=O)CN(C)C2 C(C(C)C(=O)NOCC1CC2C=CC1C2)NC(CCC1CC(OC)C1)=O C1(C)(C(=O)NCCC2OCCN(C(COCCCOC)=O)C2)CCC(C)=C(C)C1 c1(C(=O)NCCc2cn(Cc3ccccc3F)nn2)cnn2c1S(=O)(=O)NCC2 C#Cc1c[nH]nc1C(N1CCC(NC(=O)CCc2cn(C)cn2)C1)=O N1(C(C(C)Sc2ccccn2)=O)CC2CCN(C(=O)C3=CC(C)(C)C3)CC2C1 C1(C(N2CCN(CCNC(c3ccsc3Cl)=O)CC2)=O)SC2C=CC1CC2 CC(C)(C#N)CS(=O)(=O)NC(c1cnc2sccc2c1)=O C(C)(CC(C)CC(C)C)N(Cc1c(NC(=O)NCCOC)ccc(CC)c1)CC c1(C(N2CC(C)(C)C(CNC(c3ccns3)=O)C2)=O)nccc2c(Cl)cccc12 N1(C(C)=O)CC(NC(=O)CC2(n3cccc3)CCOCC2)C2(CC2)C1 C1(CC(=O)N(CCCCNC(c2csc(C(F)F)c2)=O)C)CCCCC1F c1(CCC)noc(CCCC(=O)NCC2(O)CC(NC(C3(O)COC3)=O)C2)n1 C(C(C)CC(=O)N1CC(C(C)C)C1)NC(c1cc(C)sn1)=O C(CC(=O)N(C)CC1CCCOC1)(C(C)C)NC(C(=O)NCC)=O C#Cc1ccc(C(=O)NCC(O)CN(C(=O)C#CC(C)C)C)nc1 C1(C(N(C)CC2(NC(C(C)Nc3cccnc3)=O)CC2)=O)CCCCNC1=O C1(COCC)C(C2CC2)CCN1c1nnnn1Cc1cc(Br)ccc1C N1(C(=O)CC2CCC2)CC2CC1CN2C(c1cccnc1O)=O N1(C(C=CC(C)NC(c2c(CC)c[nH]c2)=O)=O)CCCC12CCCOC2 N1(C(Cc2c(C)cccn2)=O)CCC2CCCC12C(=O)NC(C1CCOC1)C C1(C(CNC(CC2C(CC=C)C2)=O)F)CCNCC1.C(=O)CC(=C)Br C(=O)(C(CC(C)C)NC(c1cn(C(C)C)cn1)=O)N(C(COC)COC)CC c1(C(N2C(CNC(C(CC=C)(C)C)=O)CC2)=O)sc2nnc(S)n2c1C Cc1c(OCC(=O)NC2CCN(C(=O)C(F)C(F)(F)F)C2(C)C)cccc1Cl C1(CNC(C(C)OC)=O)CCC(F)(CNC(=O)C(O)Cc2ccc(F)cc2)CC1 C1(NC(c2c(C)onc2CO)=O)CCN(C(c2cc(O)no2)=O)CC1F CC1(C)CN(C(c2ccc(C(F)F)o2)C(=O)NCC2(O)CCCCC2)CCC1O N1(C2C3CN(C(C4CCC(O)C4)=O)C(C3)C2)CCc2ccccc2C1.C12CC1C2 C1(NC(C2(C)CC2)=O)Cc2ccccc2N(C(=O)CSCc2cccs2)C1 c1(C(=O)NC(CCCNC(Cc2cn(CC)nc2)=O)(C)C)ccn2nccc2n1 Cn1ncc2c(N(C3CCN(C(=O)COC(=O)CO)CC3)C)ncnc12 N1(C(=O)C=CBr)CCC2(CCCCN(C(c3cccc([N+](=O)[O-])c3F)=O)C2)C1 C12(CNC(CCNC(=O)CO)=O)CC(CNC(=O)CSC3CC3)(CO1)C2 N1(C(C2CC(=C)C2)=O)CC2(C1)SCCC2NC(c1ccncc1Br)=O C1(NC(CCn2ccc(C)n2)=O)CC2CC(C1)N(C(c1cc(O)nc(O)n1)=O)C2 CCC(CC(=O)NCc1ccc(C(=O)NCCSCC(C)C)s1)SC O=S1(=O)CCC(n2nc(C3CCCCCC3)nc2-c2ccnnc2)C1 c1(C(N2CCC(N(C(=O)CC3CCC3)C)C2)=O)ccc(F)c(F)c1 C1(CNC(C(=CC2CCCC2)C)=O)CN(C(=O)CN2CCC(O)CC2)CCN1C c1(C(N2CCC(CN(C)C(c3ccc(N)cn3)=O)C2)=O)cccc2c1CCOC2 N12CCN(C(C)(C3CC3)C1)OC2=O.c1(C(C)C)csc(C(=O)NC2CCCC2)n1 Cc1cc(C(=O)NC(C(=O)NCc2nn(C)c(=O)o2)C2CCOC2)c[nH]c1=N c1(C(=O)NCCN(C(C(C(C)C)C)=O)C2CC2)c[nH]c2cccnc2c1=O N1(C(CCn2ncc(C)c2)=O)CCN(C(=O)CCCN(C)C(C)C)CCC1C C1(CNC(C(=O)NC2CCN(C)CC2)=O)CNC(C)(C)CO1 C(=O)(CC(C)CC(F)(F)F)NCC(=C)CCNC(c1ncn(CC)n1)=O C1(NC(C(C)(F)F)=O)CC2CCC1N2C(c1ccc(Oc2ncccn2)cc1)=O Cc1cnc2c(cnn2CC(N2CC3CCN(C(C4CC4(C)C)=O)C(C3)C2)=O)c1 C(=O)(CC(C)CC(C)C)N1C(C(=O)NC(C)CC(F)F)(CC)CCC1 C(C(C)(C)CC(=O)NC1(C)CN(C(=O)Cc2cc(C)cc(Br)c2)C1)OC C1(CNC(c2cccc(Br)c2)=O)CCCC2(CN(C(C3CC=CCC3)=O)C2)O1 c1(C(N2C3CN(C(C(CCC)(C)C)=O)CC2CC3)=O)cc2c(cc1Br)OCO2 C12(C(=O)NCCCN(C3CC3)CC)CCC(C1)C(NC(=O)CCCN(C)C(C)C)C2 C1(Nc2cc(N3CCC(CSC)CC3)ncn2)CCc2cccc(Cl)c2C1 N12CC3(CC(C3)NC(C(C)C)C1=O)C2.c1(C(N(CC)CC)=O)ccc(F)c(C)c1 C1(C(N2CC(n3cccn3)(CNC(=O)CSC(C)(C)C)C2)=O)(OC)CCC(C)C1 C(=O)(C(C)(C)S(C)(=O)=O)NC1CC(C)(CNC(C(CC(C)C)O)=O)C1 N#CC1CCCN(C(C2CC3(C2)CN(C(c2cc[n+]([O-])cc2)=O)C3)=O)C1 N1(C(CCCOCC=C)=O)CCC(CNC(c2cc(C3CCC3)no2)=O)C(C)C1 C(=O)(C(F)(F)C(F)F)NCC(C)(C)NC(=O)CSCc1ccc(F)cc1 Nc1cccc(C(=O)NCCCCCCN(C(=O)C=Cc2ccccc2)CC)c1F c1(NCC2(CNC(CCC(=C)Cl)=O)CC23CCC3)ncc2cccnc2n1 Cc1csc(C=CC(=O)NC(C)CCCCNC(=O)C(c2nc(C)cs2)C)n1 S(=O)(=O)(c1cccnc1NCC1(CCCO)CC1)NCCCC(C)O C(=O)(C(C)S(=O)(=O)C(C)C)NC1(CC=C)CN(C(c2ccc(OC)nn2)=O)C1 Cc1csc(=NCC(=O)N2CC(CNC(c3ccsc3C)=O)CC23CCC3)[nH]1 N1(C(C(CSCC)NC(=O)C(C)C=O)=O)CC2CC(OC)C(C2)C1.C(=O)OC C=C=CCCC(=O)NCC(N1CCN(C(=O)CCc2cc(C)no2)CC1)C C(=O)(C(C)CC(F)F)N1CCCC(N2CCN(C(COCCC(C)C)=O)CC2)C1 C(=O)(C1CCc2nccn21)OCc1c(C(=O)OC)cccc1F N1(C(C(=O)NCCC(=O)OC)C2CCOC2)CCC2(CC1)CC(O)CO2 C=CCC(C)(C)C(=O)N1CC(C(=O)NCC2CC23CCCCC3)C(C=CC)C1 C(C)(C)(CC(=O)NC(CO)C(C)NC(C1CC(F)C(=O)N1)=O)SC CC1CCCC1C(=O)NCCCOCCN(C)C(c1nncn1C)=O C1(OC)CN(C(C)=O)CC1NC(C1OCCC1(C)C)=O.c12csc(n1)NC(=O)C2 C(=O)(C(F)C(C)CNC(c1cccc(OCC(F)F)n1)=O)N(CC)CC n1(C(C)C)ncc(C(N2CC(O)(CC(=O)N(C)CCN(C)C3CC3)C2)=O)n1 C1(NC(c2ccc(Br)cn2)C)CCNC(NC(=O)OC(C)(C)C)C1 C12(CC=C)CN(CC(c3csc(N4CC5CC4C5)n3)=O)CC(CSC3CC3)(C1)C2 CCC(O)C(C)(C)C(=O)N(CC(O)CNC(c1c(C(C)C)n[nH]c1C)=O)C C(=O)(C1CCCc2ccccc21)NCC(N(C(=O)CN1CCCC1=O)C)C1CC1 C1(CC(=O)NC2(C)CC(NC(C(C3CCC(C)CC3)CC)=O)C2)CCCCCC1 N1(C(=O)Cn2ccc3ccccc23)CC2C3CCC(C2C1)N(c1ncccn1)C3 C1(c2c(C(=O)OCC)scn2)CCCN(CN2CC(NC(C)=O)CCC2=O)C1 C12(CNC(C3CCC(C(F)(F)F)O3)=O)CC(CNC(C3(O)CC3)=O)(CO1)C2 N1(C(CCC(=O)OC)=O)CCCC(C)(C)C1CNC(C1CN2CCN1CC2)=O N1(C(=O)Nc2cnn(C3CCC3)c2)CCC12CCCOC2 C1(C2CN(C(=O)Cc3cc(F)ccc3Cl)C2)(NC(C2CCC=CCC2)=O)CC1 c1(C(N2CCCC2c2ccc(C)nc2)C(=O)NCCC)ccc(OC)nc1OC C(=O)(CS(=O)(=O)NC(C)(C)C)NCC(C)CNC(=O)C(C1CC(F)(F)C1)O N1(C(c2nc(C(C)=O)sc2)=O)CC(NC(=O)Cc2cncc(Br)c2)C(F)C1 c1(OC)ccccc1-c1noc(C2CC(NC(c3ccccc3)C(=O)OC)C2)n1 CCC(CC(=O)NCCC1(CNC(=O)CC2(O)COC(C)(C)C2)CC1)C(F)F c1(N(CCC)C(c2cc(C)ccc2Cl)=O)cc2c(nn1)CCCC2 n1(C(CC)CC)nc(C(=O)NC2CC(CCNC(c3ccoc3Cl)=O)C2)cc1C C1(CC)(CC)CC(NC(=O)COC(C)(C)CC)CN1C(=O)C(C)(C)n1ccnn1 C1(NC(c2cnc(Cl)cc2Cl)c2n(C3(C)CC3)nnn2)C2CCCCCC12 C(C(=O)NCC1CCC(C(=O)NCC2CC3CCC2C3)C1)(C(C)C)SC C1(CC(=O)NCCOC(=N)O)CCCN(C(C23CCCC2CCC3)=O)CC1 N1(C(C2CC(C)N(C)C2)=O)CC2CC(NC(c3ccn(C)c(=O)c3)=O)C(C2)C1 c1(NCCN(C)OC(N(C)C)=O)cccc(-c2ccc(C(F)F)nc2)c1 c1(C(=O)NCC23CC(NC(C4CCC4n4cccn4)=O)(C2)C3)ncccc1CO c1(C(N(C)CC2CCN(C(C3(C)CC3(Cl)Cl)=O)C2)=O)ccnc2ncnn12 C1(NC(C2(C)C(C)CN(C(C3CCCC3)=O)C2)=O)CC2CC1OC(=O)N2 C1(NC(Cc2c(OCC)cccc2)=O)CC(O)CN(C(=O)CCc2cccs2)C1 C1(CNC(C(C2CCC2)OC)=O)COCCN(C(c2ccc(F)nc2)=O)C1 CC1CC(NC(=O)C(CC2CC2)Cc2ccccc2O)CN1C(=O)C(N)=O c1(C(=O)OC)ccc(Cl)c(C(=O)NCCCN(C(C2CC3CCC23)=O)C2CC2)c1 CC1CC(=O)NCCN1C(=O)CN(C1CCC1)C(C1CCN1C)=O n1(CC)cc(C(=O)NC2CCC(C)N(C(C3CCSCC3)=O)C2)c2ccccc12 Cc1sccc1C(=O)NCCCC(=O)NCc1noc(C(N)=O)n1 N1(S(=O)(=O)CCBr)CCc2cc(-c3cc(F)ncc3O)ccc2C1 CP(C)(=O)C1CCCCCN1C(c1cc(Cl)cc(Br)c1)C(=O)NC=O C1(CNC(CCNC(C)=O)=O)CN(C(=O)C=CCO)CC2(CCC2)O1 c1(C(N2CC(NC(C3CCCC(=O)O3)=O)C2)=O)cc2c(nc1O)CCCC2O c1(C(=O)NCC2(C)CCN(C(CSC)=O)C2)ccc(C2=CCOCC2)cc1 c1(CC)nc(C(=O)NC2CCC(NC(C3(C4CCCO4)CCCC3)=O)C2)co1 Cc1ccc(CN=C(NCC(F)(F)CO)NCC2CCCCO2)c(C)c1 c1(C(=O)NCCN(C(CC)C)C)ccn2ncc(-c3ccccc3)c2n1 c1(C(=O)NC2C(CNC(C(C)NC(COC)=O)=O)CCC2)cnc(OC)cn1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CC(NC(=O)NCc2ccccc2F)C(O)C1 C1(C(C)(C)C)C(=O)N1C1CCCC1.c1(C(C)=O)cc(CCC(=O)OC(C)C)c[nH]1 c1(C(N2CC(N(C(CCC=C=C)=O)C)C3(C2)CC3)=O)cnn2c1CC(C)CC2 C(=O)(CCCCC(N)=O)NCC(C)(C)CNC(c1sccc1-c1ccccc1)=O c1(NC(CCN(C(c2c(CC)ncs2)=O)CC)=O)cccc(Cl)c1 c1(C(N2CC(COC)N(C(c3ccc(Cl)[nH]3)=O)CC2)=O)cccc2c1ncn2C C1(NC(CCOC)=O)CCN(C(c2sc(C3CCCC3)nc2C)=O)CC1F c1(C(N2CC(NC(Cc3cn(SC)nc3)=O)C2)=O)ccc2n[nH]cc2c1Cl c1(C(C(=O)NCC2C(CNC(C(COCC)C)=O)C2)(F)F)ccc(F)cc1F c1(C(=O)O)ccc(OCCOCCN(C)C(c2ccc(Cl)[nH]2)=O)cc1F.C(CF)ON.CO Cc1cc(C(=O)NC2CCN(C(c3ccc(C4CC4)s3)=O)CC2C)c(O)nn1 N1(C(CCc2c(C)noc2)=O)CC(NC(=O)C(n2cc(Cl)cn2)C)C(C)C1 C1(C(=O)NC(c2ccn(C)n2)C)CC12CN(C(c1nc(C(F)(F)F)cs1)=O)C2 c1(CCC(=O)O)ccnc(NCC(C2CCCCC2)=O)n1 C(=O)(C1CNC(=O)c2ccccc21)N1CCCC2(CN(C(C3C(C)C3)=O)C2)C1 C(CCC(=O)N1CCOCC1CCO)(C(C)C)NC(C1C(CCOC)C1)=O C1(NC(C2ON=C(C(C)C)C2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC2(CC2)C1 CCCCC(C)(C)NC(C1CN(C(=O)CC2CC3(CC3)CO2)CCO1)=O C1(O)(C(C)NC(=O)C=Cc2cscn2)CCN(C(C2(c3ncco3)CC2)=O)CC1 Cc1nc(=N)[nH]cc1C(N1C2CCC1C(NC(c1ccnn1CC(F)F)=O)C2)=O C1(Nc2nccc(C(C)C)n2)CN(C(=O)CCOCC2CCCO2)CCC1F c1(-c2c(C(=O)NC(C)C)ccnc2)nc2c(s1)CN(C(c1nc(Br)cs1)=O)CC2 C1(C(=O)NCC2CCC2)CCN(C(=O)C(O)C2CCC2)CCO1 C1(=O)C2=CCC(C2)NC(=O)C2CC(C2)N1.c1(N(C)C)cccc(C(N)=O)c1 N1(C(COC2(C#C)COC2)=O)CCCOC(CNC(c2nc(Cl)cs2)=O)C1 N1(C(C2(C)CCC(=O)CC2)=O)CC2CCN(C(C3CC3C(N)=O)=O)CC(C2)C1 N1(c2nnc(Cc3n(CC)ncn3)n2CCC(=O)OCC)CCn2cccc2C1 C(=O)(C1CCc2ccccc21)NC(C)C(C)NC(=O)C=Cc1ccc(F)c(F)c1 N1(C(CCC)=O)CCCC1CF.C1C(NC(C2COCCO2)=O)CCO1 CCC(O)(CNC(=NCCCF)NC1CCCC(C#N)C1)C(F)(F)F CCCCCC(C(=O)N(CCCNC(c1cnnc(C)c1)=O)CCO)C(C)C Cc1ccc(CNC(=O)CC2C=CC(NC(C34COCC3C4)=O)C2)nn1 C1(NC(Cn2ccc(C)n2)=O)CCC(CNC(=O)C(c2ccc(F)cc2)O)CC1 c1(C(=O)NCC(CCNC(=O)CC2CCSC2)OC)cnc[nH]c1=N C(=O)(C(F)C(C)(F)F)NC1(C(N(CC(O)CO)C)=O)CC(CO)C1 c1(CC)c(C(N2CC(CNC(c3[nH]c(C)nc3CC)=O)C3CC23)=O)cnn1C CC1(C)CCOC1CC(N1CCSCC1CCNC(c1coc(Br)n1)=O)=O N1(C(c2scc(CC)c2)C(=O)NCCN2CCOCC2)CCOCC1C#N CCC(O)C(F)(F)C(=O)NCC1(F)CCN(C(C2CCCNS2(=O)=O)=O)CC1 CC(C)CC(C(=O)N(C)Cc1cc(C(C)C)on1)N.c1(C(C#C)N(C)C)ccccc1 C(=O)(C(F)(F)C(C)O)NCC12C(CN(C(C(C(C)C)NC(C(C)C)=O)=O)C1)C2 C=CCC(CC)C(=O)NC1CC(C)(NC(c2nc(SC)ncc2N)=O)C1 c1(C(=O)NCC2(O)CN(C(CC3C(C)(C)C3)=O)C2)sccc1C#N CCCCCS(=O)(=O)CC(=O)N(CC)CC1CCCN(C(C2SCCS2)=O)C1 N1(C(CCN(CCOC)C(C2CC2OC(C)(C)C)=O)=O)CCC(CC(F)F)C1 Cc1ncn(C)c1C(N1CCOC(CCCNC(c2ccco2)=O)C1)=O c1(CC(=O)NCC2CC(C(=O)NCCCCC3CC3Cl)C2)ccc(F)cc1 C1(NC(C(CC2CC2)OC)=O)C2CC1N(C(c1ccc(Cl)cn1)=O)C2C C1(NC(=O)Cn2ccc(Br)n2)COCC1NC(C12CCC1C2)=O N1(C(c2nc(CC)oc2)=O)CCN(C(=O)CC2(C)CC2(F)Cl)C2(CCC2)C1 C1(C(=O)N(C(C)C(=O)N(C)CC2CC2(C)C)C)(CC)CCC1 CCCCC(CC)CC(=O)NCC1CN(C(C2(F)CC=CCC2)=O)CC1OCC N1(C(C2CCCN(C(C3C(C(C)C)OCC3)=O)CC2)=O)CCC(O)C(C)(O)C1 CC(C)CC(C)(C)C(=O)NCCN(C1CCCCCC1)C(C1(CF)CCC1)=O c1(NC(=O)NCC2CC(C(C)C)OCC2)cc(F)ccc1[N+](=O)[O-] c1(NC(C2CC(CNC(c3ccn(CCOC)n3)=O)C2)=O)c(Br)cnn1C C1(F)(C(=O)NCCOCCCNC(=O)C=CBr)CC12CCCCC2 c1(C(=O)OC)c(Cc2c(NC(N(CC)CC)=O)con2)cnc(C)c1O C1(NC(=O)CCF)CC2CC1CN(C(C1(c3ccccc3)CCCO1)=O)C2 c1(C(=O)NC(C(C)NC(c2c(OC)n(C)nc2)=O)C)cc(F)cc(S(N)(=O)=O)c1 c1(CNC2CC(O)(COC)C2)cccc(NC(C2CCN(C)C2)=O)c1 N(C(=NCc1ccc(C)o1)NC(C#C)C(C)OC)Cc1onc(CCCC)n1 Cc1cc(C(=O)NC(C2(O)CN(C(C3CN4CCN3CC4)=O)C2)C)c(C)cn1 c1(C(=O)NC2CC(O)(CNC(C3(C)CC(=C)C3)=O)C2)ccccc1C(C)=O c1(NCc2c(C)scc2)ccc(Cl)c(P(C)(C)=O)c1 CN1CCN(CCC(=O)N2CC(SC(F)F)C2)CC1.O=C1OCCN1CCO C1(C(=O)NCCOC)CCN(C(c2cc(Br)c(S)n2-c2ccccc2)=O)C(C)C1 c1(-c2cnc(OC)c(C(=O)Nc3ccno3)c2)ccc2c(c1)oc(=O)n2C Cc1c(NC(=O)C(C)N(C(=O)Cn2cccc2)C)cnn1C(C)C c1(OC)cc(C)cnc1C(=O)NC1(C)CC(NC(C2CCOC(=O)CC2)=O)C1 C(=O)(C1=NNC(=O)C1)NC(C)(CNC(c1cnn(C2CC2)c1)=O)Cn1cccn1 C1(C(C)NC(c2n(CCC)ccc2)=O)CCN(C(=O)CC(=O)OC(C)(C)C)CC1 N1(C(CCOCC)=O)CCN(C(C2CC3(C2)CC3F)=O)CC(O)C1 C(C(C)C(C)(F)F)N(C(C(C)CN(C)C)=O)C1C=CCCC1 S(=O)(=O)(c1c(OC(F)(F)F)cccc1OC(F)(F)F)N1C(C)CCC(O)C1 c1(CN(C(CCN(CC#C)C(c2nocc2Cl)=O)=O)C)ccc(C)cc1 C1(CNC(=O)CCC2CCC2)CCC(CNC(C23CC(CO2)C3)=O)CC1 N1(C(c2nc(-c3ccn(C)n3)sc2)=O)CCCCC2CCCCC12 Cc1ccc(NC(=O)C(N2C(C(F)(F)F)COCC2C)=O)cc1Cl c1(C(N2CC(C)(NC(C(C(C)C)OC)=O)C2)=O)cc2ccccc2o1 C12(NC(=O)CCCc3ccsc3)CCN(C(=O)CCOCC3CC3)CCC1C2 C=CC1CN(C(c2csc(C3CCCCC3)c2)=O)CC1NC(=O)C#CC1CC1 C1(CC(N2CCC(Cn3cc(CC(COCC)O)nn3)C2)=O)CC2(CCCC2)CO1 N1(C(c2ccc(O)nc2)=O)CCC2(CCC(N3CCCCCC3)CC2)CC1 N1(C(c2cc(C)sc2Br)=O)CCN(C(=O)CCCN(C)C)CC1CF C12(C(=O)NC(CCC)CC)CCC(CC1)N(C(C1CC3(CCC3O)C1)=O)C2 c1(OC)cc(N)c(C(=O)NC(C)C(C)NC(c2cc(Cl)sc2Cl)=O)cc1F c1(C(C)NCC2(C(=O)Nc3cc(SC)n[nH]3)CC2)ncc(Br)nn1 c1(CNC(C2(CC=C)CCC2)=O)ccc(C(=O)N(CCC)CCO)s1 c1(NCC(F)(F)F)ccccc1OC.C1(NC2(C)c3nnnn32)CCCCC1.C1COC1 C1(C)(OC)CC2CC1CC2NC(=O)CNC(=O)Cc1ccc(CN)cc1[N+](=O)[O-] N1(C(=O)CC2CN(C(c3cc(O)cc(Br)c3)=O)CCO2)CCN2CC(O)CC2C1 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC)(CC)NC(C(C)OCCOC)=O c1(C(N2CC=CC2CF)=O)ncc2ccccn12.C#CC1(CO)CCN(C(N(C)C)=O)C1 c1(CC(C(=O)N(CCCNC(=O)C(C)O)CC)C)ccc(OC)cc1 S(=O)(=O)(C1CC2(CCC2)C1)NC(c1ncc(C(=O)OCC)nc1)=O CC(C)CC(C)(CNC(=O)CCc1ccsc1Cl)NC(C1CCOC1)=O N1(C(c2n(COC)ncc2)=O)CCOC(CNC(=O)C(O)C2CCC2)C1 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC(=O)NC(Cn1ncc(C)c1)C)O c1(CN(C(CC(=C)C)CO)C2(n3nnnc3S)CCSCC2)c(Cl)cccc1Cl N1(C(c2c(CC)cccn2)=O)CCC(NC(c2sccc2CO)=O)C(C)C1 N1(C(CCNC(=O)NC)=O)CCN(CCN(C(=O)CC2CCCC2(F)F)C)CC1 c1(N(CCCn2ccnc2)C)nc2cc[nH]c2c(=NC2CC(n3ccnc3)C2)[nH]1 C1(C(=O)NC(C2(O)CN(C(c3csc(F)c3)=O)C2)C(C)C)(C(F)F)CC2(CC2)C1 C12(CNC(C(C)(C3CCOCC3)OC)=O)CC(C1)C(NC(C1(SC)CC1)=O)CO2 N1(C(c2nccc(CC)c2)=O)CC2CCN(Cc3ccc4cc[nH]c4n3)CC2C1 N1(C(c2c(C(=O)OC)c[nH]n2)=O)CC2CCC(C1)C2NC(C12CC(F)(C1)C2)=O c1(OC)cc(N)c(C(N2CCC2CNC(C2CC(O)C2)=O)=O)cc1Br CCC(C)(O)C(=O)NCC(C)(O)CNC(=O)CC(=O)OC(C)(C)C CCCCC(C(=O)NCC1CCCC1NC(c1cc(Cl)no1)=O)NC(N)=O Cc1ccc(Cl)c(OCC(=O)NC(C)(CNC(C23CC(C)C2C3)=O)CO)c1 C1(CNC(CCSCC)=O)CN(C(=O)CSc2nnnn2C)CC12CCC2 c1(NC(C)CNC(c2ccon2)=O)ncc(Br)cc1C#N c1(C2(C(=O)NC3C(NC(COCC#C)=O)CC3)CC2)ccc(OC(F)F)cc1 N1(C(C2C(CC)CCCC2)=O)CC2(CO)CC1(C(=O)NCc1ccn(C)n1)C2 N=c1[nH]c2ccc(C(N3CCN(C(=O)C(O)C4CC4)C4CCC34)=O)cc2s1 C1(F)(CN)CCN(C(=O)Cc2cc(F)cc(I)c2)CC1 C1(C(=O)NCC2CCN(C(CC3(COC)CC3)=O)C2)CCCOC1C C(=O)(C1=C(Cl)CC1)NC(CNC(=O)CCc1ccc(Cl)s1)CO c1(C(N2CC(NC(C(C)OCC=C)=O)C(SC)C2)=O)ccc2scnc2c1 C1(OC)CCCCC1C(=O)N(C)CC1COCCN1C(=O)CC1CCC1 CC1(O)COCCN(C(C2CCCCN2C(=O)CSc2cc(F)cc(F)c2)=O)C1 c1(C(=O)NC2CN(C(c3ncc(CC)nc3)=O)C(C)C2)cc(C)c(C)cc1N c1(CNC2C(C(=O)Nc3onc(C)c3Br)C2)ccc(Cl)c(F)c1 N1(C(C(c2ccc(Cl)c(Cl)c2)C)=O)CC2(C1)CN(C(=O)Cc1cnsc1)C2 S(=O)(=O)(c1cccc(NC(=O)N(C)CC2(OON)CCSCC2)c1)NCC.CC C(C(O)CN=c1ncnc2[nH][nH]c(C)c1-2)NC(C(CCC)OCC)=O c1(OC)ncc(Cl)c(=NCC2CC(C)N(C(c3cc4n(n3)C(C)CCC4)=O)C2)[nH]1 N1(C(C(C2CCCC2)OCC)=O)CC2CC1C2NC(=O)CCF c1(C(=O)NC2(C)CCCN(C(c3cccc(N)c3F)=O)C2)cnn2cccnc12 N1(C(c2ncn(C3CCN(CC)CC3)c2)=O)CC(C)N(C(=O)OC)CC1C CCCCCC(C(=O)NN(C1CCC2(CC1)CC2CO)CC)N1C2CCCC1CC2 C1(NC(c2cnc(O)[nH]2)=O)CCN(C(=O)COC(F)F)C1c1ccccc1 CCCC(C(=O)N1CCN(C(=O)Cc2cncnc2)C(CC2CC2)C1)C(C)C c1(C(=O)NC2(C)CN(C(C3COC(=O)N3)=O)C2)cccc(C(N)=O)c1N c1(OC)ccccc1C(N1CCC(C(N2CCN(CC(=O)O)CC2)=O)CC1)=O Cc1cc(Cl)cc(C)c1C(=O)NC1CCCN(C(C2CCNC2=O)=O)C1 CC(C)C(C(=O)Nc1ccccc1Br)OC(=O)CCCc1cnn[nH]1 C(CC(C)C(=O)NCCCCN(C)C(C1CC(O)CN1C(C)=O)=O)OC c1(C(=O)N(C2C=CCCC2)Cc2ccc(I)cc2)ccc([N+](=O)[O-])o1 c1(OC)c(C)cnc(C(C)NC2CCc3ccccc3C2)c1C c1(C(=O)NC(C(C)NC(=O)Cn2nnc(=O)[nH]2)CO)ccc2c(c1)OCC2 N1(C(C(CC2CN(C(=O)Cc3cocn3)C2)F)=O)CC(C2CCCCC2)C1 C1(CC=C)(C(=O)N(C(CCC)C2CCC2)CC)CCCN1C(=O)Cc1cccnc1C c1(C(N(C)CC2CCN(C(C3CC3F)=O)CC2)=O)ccc2nsnc2c1 N1(C(c2cc(CCOC)on2)C(=O)NCCOCC)CCC2(C1)OCCO2 O=S1(=O)CCC(c2noc(-c3cnc(-c4cscc4Cl)cn3)n2)CC1 Cc1ccccc1CS(=O)(=O)N(C)C.c12c[nH]nc1C(=O)N2 Cn1cccc(C(N2CCC(O)(CC(=O)NCC3(CO)CCOC3)C2)=O)c1=O C1(CNC(CN(CC)CC)=O)Cc2ccccc2CN1C(c1n[nH]cc1OC)=O c1(C(=O)NC(C2CN(C(c3ncc(CC)nc3)=O)C2)C)ccc2scc(C)c2c1 CN1CCN(C)CC(C(N2CCC(CCNC(c3cn(C)ccc3=O)=O)C2)=O)C1 N1(C(C(N=S(C)(C)=O)=O)=O)CC2(CCCC2N=c2ccnc(C(F)(F)F)[nH]2)C1 C(=O)(C(C)(C)C(=O)NC(CNC(C1(C)CNC(=O)C1)=O)C1CCC1)OCC N1(C(c2cc(C(C)=O)[nH]n2)=O)Cc2ccnn2CC(NC(=O)C(O)CN(C)C)C1 c1(C(=O)NCC2CCC(C(N3CC=CC3(C)CO)=O)O2)cc([N+](=O)[O-])c[nH]1 CC(C)C(C)(CNC(c1cc[nH]c1)=O)NC(=O)C(C)n1ccnc1 CCCC(C(O)C(=O)N1CC=CC1CN(C)C)NC(c1snnc1C)=O Cc1ccnnc1C(=O)NCC1(C)CCN(C(c2ccc(F)s2)=O)C1 CCCCC(=O)NC(Cc1cn(Cc2cnn(C3CCC3)c2)nn1)C(=O)NC CCCC(CC)CC(=O)N(CC(O)CN(C(=O)Cc1ccc(OCC)cc1)C)C c1(C(N(C(C)C(=O)O)CC)=O)cc2c(C)cc(C(=O)OC)cc2[nH]1 C1(N(C(CCC(=C)C)=O)C)CCN(C(=O)Cc2ccc(O)cc2Cl)CC12CC2 O=C1CCC(C(=O)NCC2CCCN2C(c2cc(C3CCC3)on2)=O)C1 N12CCC(CC1)S2.C1(C(C)=O)(C(=O)N(C)CCN(C)C(C2(CCO)CC2)=O)CC1 Cc1oc(CO)cc1C(=O)NCC(C)(O)CNC(=O)Cn1cccn1 N1(CCC(=O)NC(CNC(C)=O)(C)C)CC(C(F)(F)F)CCC1C(F)(F)F C#Cc1cc(F)c(C(=O)NC2(CC=C)CCN(C(C3CC(C)=NO3)=O)C2)cc1F Cc1cc(N2CCC3NCCC3C2)nc(=NCc2nc(C(F)(F)F)cs2)[nH]1 C1(F)(CNC(C(C=CC)O)=O)CCC(CNC(c2c(C)noc2C2CC2)=O)C1 c1(C(=O)OC)cc(-c2cn(CCCN(C)C(c3nc[nH]n3)=O)nn2)cs1 N1(C(C(CC)OCC)=O)CCC(C)C(NC(C2CC(=O)N(CC3CC3)C2)=O)C1C c1(C(N2CCC(C)(C(=O)Nc3c(Br)ccc(C)n3)C2)=O)c(C)cc(Br)cc1F C#Cc1cnn(C)c1C(=O)NCC1CC(NC(=O)CSc2ncccc2O)C1.CC Cc1ccc2c(c1)CC(C(=O)NC1CC1CNC(c1cccn(C)c1=O)=O)S2 CCCC(C)CCCC(=O)NCCN(C)C(C1(CO)CCOCC1)=O C(=O)(C(C)(F)C(F)(F)F)NCC(C)N(C(c1c(C)[nH]c(C)c1C)=O)C C1(NC(c2c(C)nc(C)[nH]2)=O)CN(C(=O)Cc2ccnn2C2CCC2)CCC1F C#Cc1ccc(C(=O)NCCC2CC(F)(F)CN2C(c2occc2CC)=O)cc1 C(C(F)(C(=O)NCc1cccnc1)C(C)C)NC(c1[nH]cc(C)c1C)=O C(CC(C(N)=O)NC(=O)C(C1(O)CCCCC1)NC(=O)CCOCC(C)C)OC CC(CCC(=O)NC(C1CCN(C)CC1)C)NC(c1cc(C2CC2)no1)=O C12(C(N3CC4C(CC(=O)NC(C5CCOC5)C#C)C4C3)=O)CCCC1C2(F)F CN1CCN(CC(=O)NCC(c2ccccc2)NC(=O)Cc2nccn2C)CC1 C12(C(N(C(CC)C3CC3)C)=O)CCC(NC(C3CCOCC3(C)C)=O)(CC1)C2 Cc1c(C(c2nnnn2CC(F)F)NCc2ccnc(Br)c2F)cccc1F C1(CC(=O)NCC(CC)(C)NC(c2ccc(CO)c(F)c2)=O)CC(O)C12CCC2 Cn1nnc(CNC(=O)CC2(C)OCCO2)c1C(N1CCOCC1)=O c1(CC(=O)NCC(C)CN(C)C(c2cn(C)nc2O)=O)ccc2c(c1)CCOC2 n1(CC(=O)OC2CC(OCC)C2(COC)CC)cccc(N)c1=O c1(C(NOC(C(=O)N2C(C(C)(C)OC)CCC2)CC)=O)cc(C#N)c[nH]1 N1(C(CC2(OC)CCCCC2)=O)CC(CNC(=O)C=Cc2ccnn2C)C2(CC2)C1 c1(CNC2(c3n(CCCSC)nnn3)CC(Br)C2)nn(C)nc1Br c1(C(=O)NCC23C(CN(C(C4N(CCC)CCC4)=O)C2)C3)c(C)cc(Cl)cc1C N1(C(c2nc(CC)oc2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC(C1)O2 CCC(C(=O)N(CC(=O)NC(CC1CC1)C(=O)OC)CCO)OC c1(CC(N2CCC(N(C(Cc3nnc(C)s3)=O)C)CC2)=O)cc(O)nnc1O N1(c2ncc(C(=O)OCC)cn2)CCCC(C2CC2NC(=O)CSCC(N)=O)C1 C1(C(N(C2CC(OC)C2)C)=O)CN(C(C2CCCCC2(C)C)=O)C2(CCC2)C1 N#Cc1c[nH]c(C(=O)NCC2CC2NC(C2CC2C(N)=O)=O)c1 C(=O)(CCCC(CC)NC(c1cnnc(O)c1)=O)NCC(C)OCC=C N1(C(C2(OC)CCCCC2)=O)CC(NC(=O)NCCC(=O)NCC)C(C)(C)C1 CC1=NC(C)(CNC(=O)C(CCC2CC2)NC(c2sc(F)cc2C)=O)CS1 C12(CNC(C(COC)(C)C)=O)CCC1CCN2C(=O)CCCc1nc(C)no1 C(=O)(CCC(C)CCCC)NC(C1CCCC1)CNC(C(C=C)CC)=O C(c1ccc(Br)o1)=C(C)C(N1CCN(C(C)(C)C)CC1)=O.C(=O)C=CCF c1(CCC(C)=O)ccc(C(N2CCSC(C(=O)OC(C)(C)C)C2)=O)cc1 c1(C(N2CCCC(N(C(C3ON=C(CC)C3)=O)C)C2)=O)cccc2c1CCCN2 N1(C(C2CCN(C)C2)=O)CCCC2CN(C(=O)Cc3cc[nH]n3)CC12 c1(C(N(CC(C)NC(=O)COCCCOC)CC)=O)cc2ccccc2cn1 C12(C(N(CCC(C(C)C)NC(=O)C(C)(F)F)C)=O)CCCC1C2(F)F C1(CC)CCCC1C(N1CC(NC(c2cnn(C3CCOCC3)c2)=O)C1)=O CC1=NOC(C(=O)NC(C)CCCNC(=O)C=CBr)C1 N1(C(c2n(CC)ccn2)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)C(C)C1 CS(=O)(=O)c1ccc(C(=O)NCC2CCC2NC(=O)Cc2cccnc2Cl)[nH]1 C1(OC)CN(C(c2cn(C3CC3)nn2)=O)CC1NC(C1CCC1(OC)OC)=O c1(C(=O)NCC(C2CCCCC2)NC(C2C(C)C2C)=O)cnc2nccn2c1 n1(CC)cc(C(N2CCCC(CN(C)C(C3CC3(F)F)=O)C2)=O)c(C(C)C)n1 CC1CC(NC(c2coc(C3CC3)n2)=O)CCN1C(C12CCC(C1)OC2)=O C(=O)(C#CC(C)(C)CNC(c1oc(CO)cc1C)=O)NCC(C1CCCC1)OC N1(C(C(C2CN(C(C3CNC(=O)C3)=O)C2)OC)=O)CCC(CO)C(O)C1 C(=O)(C1CSc2ccccc21)N1C(CN(C(CC2C(C)C(=O)CC2)=O)C)CCC1 C(c1cnc[nH]1)=C(C)C(=O)N(C(CNC(=O)Cc1csc(C(C)C)n1)C1CC1)C C1(C(N2CC(O)(CNC(Cn3ccc(C)n3)=O)C2)=O)CCN(C2CC2)C1=O Cc1cccnc1CC(N1CCC(CN(C(=O)CN2CC(C)(C)C2)C)C1)=O CC1(C)CC(CC(=O)NCC23CC(CN2C(c2n[nH]cc2C2CC2)=O)C3)CO1 c1(CC(C(=O)NCC=CCNC(C2C(C=C)C2)=O)O)ccccc1Cl Cc1ccc([N+](=O)[O-])c(C(=O)NC(C)CN(C)C(c2cc(Cl)c(Cl)cc2N)=O)c1 C1(CC)CN(C(c2cn(C3CC3)nn2)=O)CCN1C(c1nn(C)c(N)c1C)=O c1(C(C(=O)NCc2cccs2)N(C(CSC)C)C)ccc(Cl)o1 C(C1=CCCN(C(c2c(C)cncc2C)=O)C1)NC(C(CC)NC(N)=O)=O Cc1cnc(C(=O)OC2CCN(C(=O)OC(C)(C)C)CC2F)cc1C CN=c1nc(C(=O)NC2CC(CNC(C)=O)CN2C(=O)OC(C)(C)C)cc(C)[nH]1 C(=O)(CC(C(F)(F)F)NC(=O)CC(C)(C)C)N1C(C(=O)OC)CCCC1 c1(NC(=O)NCC(CC(C)C)N(C)C)ccc(F)c2c1CNC2 c1(C(=O)NC2(CC=CC(=O)OCC3COCCO3)CCC2)ccc(Cl)cn1 CN=c1ccc(C(N2CC3(CC3)CC2C(=O)Nc2ccc(F)cc2O)=O)c[nH]1 c1(-c2cn(CC(=O)OCC)nn2)cccc(NC2CCNCC2)c1 C1(C(=O)NC(c2cccc(OC)c2)COC)COCCN(c2cc(O)nc(C)n2)C1 N1(c2n(CCOCCOC)c(C3(C)CCCCO3)nn2)CC2OC(C)(C)OC2C1 C1(NC(C(c2ccccc2Cl)(C)C)=O)CN(C(C2CC=CCC2)=O)CC1O C1(c2nc(C)on2)CCN(CC(O)CC(=O)C(c2cccc(Br)n2)(F)F)CC1 N1(C(C(C)OCCCC)=O)C(C(=O)NCC(C)(C)CCOC)CCC1C C1(NC(C2C(CNC(CN3C(C)CCC3)=O)CCCC2)=O)CCC2(CC1)N=N2 CCC(CC(=O)NC1CN(C(c2cccc[n+]2[O-])=O)C2(CCC2)C1)C(C)(C)C CC1CC(NC(=O)C2CC2)CN1C(=O)CCc1ccc(F)cc1 C(C(C)(C)C(=O)N1CC2C(NC(=O)COc3ccccc3)C2C1)NC(C)=O C#CC1CN(C(=O)C(Cc2cc[nH]n2)NC(=O)Cn2cnnc2)CC1O c1(OC)c(-n2cc(C(C)NC(CC(O)CC(C)C)=O)nn2)cccc1F N1(C(C(=O)NCCCC)C2CC=CC2)CCN(Cc2ccon2)CC1 N1(C(C(CCF)NC(Cn2c(C)ccn2)=O)=O)CCC2(C=CCO2)CC1 c1(CC(=O)NCCCCNC(=O)CC23CCCC2C3)ccc(OC(F)F)nc1 C1(C(N(C)Cc2n(CC)ccn2)=O)CC(NC(=O)C=CC2CCCC2)CCO1 c1(-c2cccc(CC)c2C)cccc2[nH]nc(C(=O)NC3CCC(F)(F)C3)c12 c1(C(N2CC3(C(C(N4CCC(C)(C(=O)OC)C4)=O)C3)C2)=O)c(F)cc(Cl)cc1F N1(C(Cn2cc(CNC(COCC#C)=O)nn2)=O)CCC2(CC1)CC2C#N C(=O)(C1=C(Cl)CCCC1)NCCC1(C(N2C(CC)CC(O)C2)=O)CCCC1 c1(N2CC(OCCNC(CC(C=C)c3ccccc3)=O)C2)ncnc(Cl)c1Br C1(OC)CC(CO)N(C(c2ccccc2CNC(c2cncs2)=O)=O)C1 O=C(NN1CCCC1C(=O)Nc1cncnc1O)C1=CC2(CCOCC2)C1 Cc1[nH]nc(C(N2CCCC(CN(C)C(C3CC3F)=O)C2)=O)c1Br Cn1nc(C(=O)NC2(NC(=O)COCCc3nccn3C(C)(C)C)CCC2)cc1Cl Cc1cc(C(=O)N(C)CC2(O)CN(C(=O)C(F)(F)CC3CC3)C2)c(N)c(Cl)n1 c1(CC(=O)NC2CC(CNC(=O)CCC3CCCCC3)C2)cccc(O)n1 C1(N(C(=O)C(C)(C)OCC(F)(F)F)C)CCn2ccnc2C1 C(=O)(C(CC#CC)NC(=O)C(F)C(C)(F)F)NC1(C)CC(=C)C1 c1(C(N2CC(NC(C(CC)SC)=O)C(O)CC2)=O)ccc2cnccc2n1 Cc1cc(-c2ccc(CNC(c3ccnc(Br)c3)=O)cn2)cc(C)n1 C(CC(C)C)(CC(C)C)NC(CC(CC)NC(C1C(=C)C1)=O)=O CCCCCCCC(C)NC(C)C(=O)NCc1c(C)cc(C(=O)O)c(C)c1C Cc1ccc(C(N2CCCN(C(C3CNC(=O)C3)=O)CC2C)=O)c(N)c1C C(C(=O)C1CCCc2ccccc21)C(NNC(c1ccc(C#N)cc1Br)=O)=O c1(C(N2CCN(C(C3C(=C)C3)=O)C(C3CC3)C2)=O)cc(C)c(F)cc1Cl C1(C(=O)OC)C(O)CCCN1Cc1cccnc1N1CCOCC1 C1(NC(C2(C(=O)NC)CCC2)=O)CCC(C)(CNC(c2c(C)nsc2C)=O)C1 C1(NC(Cn2c(C)cnc2)=O)CCCN(C(=O)CCc2ccc(Cl)nc2)C1C Cc1ccc(OCCC(=O)NCC(C)NC(c2nccnc2N)=O)c(Br)c1 N1(C(C2(C)CCC(=O)NC2)=O)CC2CN(C(C3CC(=O)C3C(C)(C)C)=O)CC2C1 C(C(C(=O)NC1CCCCN(C(=O)C2=CCCC2)C1)C(C)(C)C)OCC=C CCCCC(O)CC(=O)N(CC(C)NC(c1cnc(OCCOC)c(Cl)c1)=O)C C1(CC(=O)NCc2c(CCNC(C=C=C(C)C)=O)ocn2)CCC(F)(F)CO1 C#Cc1cncc(C(=O)NC(c2cnn(C)c2)C(=O)NC(CC)C(C)(F)F)c1 c1(C(=O)NC(c2nncs2)C)cccnc1CNC(=O)CCCF N1(C(=O)CC2C3CCCC3N2C(=O)CCC2CC2C#N)CC2(CNC(=O)OC2)C1 CCCCCCCCOCC(=O)N(C1CN(C(c2ncn(CC)n2)=O)CC1F)C CC1OC2(C)CCC1(NCc1sccc1Br)CC2 N1(C(c2ccc(C)s2)=O)CCC2C1CCCN2C(c1ncc(Cl)cc1C)=O c1(NCc2ccc(-n3c(C)ncn3)cc2)ncnc(Nc2ncc(F)cc2Br)c1C N1(C(c2c[nH]c(=N)s2)=O)CCC(O)C(C(=O)Nc2ccn3nccc3c2)C1 N1(C(CC2N(C)CCC2)=O)CCSCC1C(=O)N(CC(c1nn[nH]n1)C)C N1(C(CCSCC(C)C)=O)CCC2CCN(C(=O)C=C(Cl)Cl)CC2C1 c1(CN2C(C(=O)Nc3ccc(C(=O)OC)nc3)CC(C)C2)cccc(C)c1O C1(F)(CNC(CC=CC)=O)CCCN(C(=O)CN(CCOC(C)(C)C)CC)C1.C1CC1 c1(C(N(CC(CN(C(=O)C(F)=CCCF)C)O)C)=O)cccc(-c2cccs2)n1 c1(C(=O)NCCN(C)C(C2CCC2F)=O)ccc2c(c1)CCNC2=O N1(C(COCCC=C)=O)CC(n2cc(-c3ccncc3Cl)nn2)C(C)C1 C1(C(=O)NC(COC)C(C)C)CCN(C(=O)CN2CCNC(=O)C2)CC1(C)C CCC(C)CCCCC(=O)NCC(O)CN(C(=O)Cc1conc1C)C Cn1[nH]c(=NC(=O)CN2CCCC(O)CC2)cc1-c1nn[nH]n1 CC(F)(F)CCC(=O)NCc1cc(C(=O)NCCCC(O)CO)n[nH]1 C1(C(N(C)CCN2CCCC2=O)=O)CCN(S(=O)(=O)CC2CC2)CC1 Cc1cnc(CN2CCC(C(=O)NCc3cn[nH]c3)C(O)C2)c(C)c1 c1(C(=O)NC(C2CN(C(c3ccncn3)=O)C2)C)cnc(O)n(C)c1=O C1(NC(C#C)=O)CC2(C1)CN(Cc1cc(Br)cc(I)c1)C2 CC1CCC(C(N2CCC(C)(CC(=O)NCC3CCCCS3)C2)=O)CC1 N1(C(Cc2c(C)occ2)=O)CC2CCN(C(=O)CC3(C)CCCO3)C2C1 Cc1ccc(Br)c(C(=O)NCC23CC2CN(c2nccc(C(F)(F)F)n2)C3)c1 C1(NC(CN(S(C)(=O)=O)C)=O)CCN(C(=O)COc2ccc(F)cc2)CC1(C)C C=CCC(C)(CC)C(=O)NCC1CCCN1C(=O)Cn1nc(C)nc1C Cc1c([N+](=O)[O-])ccc(NCC(c2cc(F)cc(F)c2)C)c1[N+](=O)[O-] C1(C(=O)OC)C(OC)C(OC)CN1CC(c1sc(C(C)(C)C)nc1C)=O c1(CC(C)NC(c2n(CC=C)nnn2)C=Cc2ccccc2)ccc(C#N)cc1 c1(OC)cccc(CC(=O)C(=O)NC2CC(CNC(c3cnc(C)[nH]3)=O)C2)c1 N1(C(c2[nH]c(C)c(C(=O)OC)c2C)C)CC2(CC(C(=O)OCCSCC)CO2)C1 c1(CC)oc(C)cc1C(=O)NCCCN(C)C(C1(OC)CCCCC1)=O c1(C(C(=O)NCCOCCCNC(c2cnco2)=O)(F)F)ccc(F)cc1F c1(C(NC(NCC(C=C)(F)F)=S)C)ccc(Cl)cc1Cl C1(C)(C(N2CC(SC)C(NC(c3cc(O)cs3)=O)C2)=O)CCCC1(F)F CC1(C)CC(=O)N(CC(N2CC(NC(=O)Cc3ccnc(O)c3)C2)=O)O1 C1(NC(CCCCCC)=O)CCCC12CN(C(c1cc(O)ccc1O)=O)C2 C(CC(=O)NCC(Cl)Cl)(C(F)F)NC(C(CC)=COC)=O C(=O)(C#CC1(C)CC1)NC(CCC)C(=O)N1CCN(C(=O)C(C)SC)CC1 CC(C)C(C)CC(=O)NCC(CC1CC1)C(=O)NC1(c2nc[nH]n2)CC1 Cc1cncc(C(=O)NC(CNC(=O)C(=O)N(C)C)C(C)(C)C)n1 C1(Cn2cc(CC(C)O)nn2)CCN(C(c2cc(O)nc(O)n2)=O)CC1(F)F c1(CNC(NC(C)C)=NCc2cc(Br)c(F)cc2F)ccc2c(c1)OCCO2 Cc1oc(CNC(=O)C(C)(C)C2CCC2)nc1C(=O)Nc1cncc(N(C)C)c1 N1(C(CCOCC(C)C)=O)CC2(CCC(C(=O)NC3CC3CC(C)(C)C)O2)C1 C(=O)(CCC1=NNC(=O)CC1)NC1CC(NC(c2cc(OC)no2)=O)C1 C1(C(=O)NC2(CNC(C3N(C)C(=O)NC3)=O)CCC2)CCC2(CC1)COCCO2 c1(SC)ccc(C(=O)NC2(C)CN(C(=O)CC3CC(C)=NO3)C2)s1 N1(C(c2nc(C)oc2)=O)CCC2(CC1)CC2C(=O)Nc1ccc(O)cc1Br c1(C(N2CCC(O)(CNC(c3cnc(CC)o3)=O)C2)=O)cnc2[nH]ncc2c1 C1(Cc2cn(C(CNC(C3(C=C)CCC3)=O)C)nn2)CC2CCC1CC2 C1(C)(NC(CC(C)n2ccnc2)=O)CCCN(c2ccc(CO)cn2)C1 c1(C(N2CC3C(CNC(C45CC(C)(C4)C5)=O)(C3)C2)=O)cccc(=S)n1O C#CC1(NC(C2C(CNC(C3CCCCS3)=O)C2(C)C)=O)CCCCC1 CC(C)(O)C(C(=O)N1CCC(c2ccco2)C1)NC(=O)CCOC1CC1 Cc1noc(C)c1CNC(=O)CC1(CN)CC1.C(=O)(C(C)C(=O)OC(C)(C)C)NC.S C1(NC(CC)=O)CS(=O)(=O)CC1NC(c1nn(C(C)(C)C)cc1Br)=O C=C(C)C1OCCC1CNC(=O)CC(C)(C)N(C)C(c1ccc(Cl)o1)=O Cc1nn(C)c(C)c1CCC(=O)NC1CC1NC(=O)CNC(C1CCC1)=O.C1(S)CC1 C1(CNC(c2c(COC)ccs2)=O)CN(C)CCN1C(C1CCOC1C)=O c1(OCC)nc(Cl)ccc1C(=O)NC1CCC(NC(c2c(C)ncnc2O)=O)C1 N1(C(C)=O)CCC2(COC(CNC(c3cc(C(F)F)[nH]n3)=O)C2)C1 c1(C(N(C(C(C)O)=O)C)C)cn(CC2(COCC3CC3)CC2)nn1 c1(C(N(C)CC2CCCN(c3nc(C4CC4)ns3)C2)=O)cnc2c(Cl)cccn12 C(C(COC)C(=O)N(CCCNC(c1cn(C)nc1Cl)=O)C1CC1)OC c1(C(N2C(CNC(C3(O)CCSC3)=O)CC3CCCC23)=O)cncc2c1CCC2 Cc1nc(CNC(=O)CCc2nccs2)oc1C(=O)NC(C1CC2(CCC2)C1)CO C1(C(=O)NCC(C)(C)C(N)=O)(CC)CCN(C(=O)C(C)C(C)n2cccn2)CC1 c1(NC(CCCC)CCC)ccc(S(=O)(=O)NCCS(=O)CC(F)(F)F)cc1F O(C1CCCCc2ccccc21)C(c1cn(C)[nH]c1=N)=O C(=O)(C(C)(C)C(N)=O)NC(C(=O)NCC=CCSC)Cc1ccoc1 C(=O)(C1=NOC2COCC12)NC(CCCC)CNC(c1onc(C)c1C)=O c1(NCC)cc(Cl)ccc1C(=O)Nc1cc(-c2ccccc2Br)no1 c1(C(=O)NC2C=CC(CNC(C)=O)C2)ccc2c(c1)CC(=O)N2 C1(C(=O)NC2(c3cncs3)CC2)CN(C(=O)Cn2ccccc2=O)CCO1 C1(N=[N+]=[N-])(C(=O)NCC2CC(CNC(C(=O)NC(C)C)=O)C2)CC1 c1(C(=O)NC(CCN(C(C)=O)C)C(C)C)cc2ccc(O)cc2[nH]1 C1(NC(C(=O)N(CCCn2ccnc2)C)=O)COCC1N1CCOCC1 C12CC3(C1)CN(C3)C2=O.c1(NS(CC#N)(=O)=O)c(Cl)ccnc1Br N1(C(C(c2ccccc2)C)=O)CC(C(=O)Nc2ccccc2C#N)C(C)(C)C1 C1(CNCC2CCCC(OC)C2)Cc2cc(F)ccc2NC1=O c1(C(=O)NC2CCC(NC(c3cc(CC)on3)=O)C2)cn(C)c2ccc(F)cc12 C1(C(=O)OC)CN(C(=O)CC2CCCC2)CC1NC(=O)CCC(C)SC(C)(C)C c1(C(N2CC(CNC(=O)CCC3NC(=O)NC3=O)OCC2)=O)cc(Cl)nnc1O N1(C(c2cc(OC)cc(C)c2)=O)CC(C)OC(C)(c2ccccc2)C1.c1(C)cccs1 N1(C(c2c(C)noc2C)=O)CCC(C2CC2)(NC(c2cnc(CC(C)C)[nH]2)=O)C1 C(=O)(C(C)CN(C)C)N(CCCNC(CC=C(C)C)=O)CCO c1(C(C(=O)N(C)CC2(CNC(=O)C=Cc3cnc[nH]3)CC2)(F)F)ccccc1C#N Cc1n[nH]c(C)c1N(C(=O)C(C)N(C)C)N(C)CCNC(=O)C(C)(C)C CCCC(C(=O)NCc1c(C(=O)NCCCn2cnnc2)c[nH]n1)OC N1(C(C(C)NC(CC)(C)C)=O)CC(C(=O)NC2CC=C(C)CC2)C(C)(C)C1 N1(C(=O)OC(C)(C)C)CCC2(CCOCC2)C1C(=O)Oc1[nH]nc([N+](=O)[O-])c1Cl c1(-c2c(C)csc2C)ccc2c(c1)CCN(C(c1cc3n(n1)CCCNC3)=O)C2 c1(NC(c2cc3ccncc3[nH]2)=O)cccc(S(=O)(=O)O)c1.C12(O)CCN(C1)C2 C12CCCCN1C2=O.C1(C(=O)NCCN(C(=O)OC)C)CCC[SH]1CC(=O)OC c1(SC)cc(C(N2CC(CNC(C3CC3C)=O)C3CC23)=O)oc1C C#CC1(C(=O)NC(C)Cc2ccco2)CN(C(c2cc[nH]c2)=O)C1 c1(CNC(C2N(C(C)=O)CSC2)=O)cc(Cl)ccc1F.C123CC(C1)(C2)C(=O)NC3 N1(C(C(C)NC(CC)=O)=O)CCC(NC(=O)Cc2cnc[nH]2)C1 Cc1nn(C)cc1C(=O)NCC1(NC(C2CN(CC(C)C)C2)=O)CC1 c1(C(N(CC(CNC(C2C(C)C2C)=O)C)C)=O)ccc(-c2cnnn2C)cc1 c1(CC(=O)NC2C(NC(Cn3cnc(C#N)n3)=O)CC2)cccc2[nH]ncc12 N1(C(C2(CC)COC2)=O)CCC(C)(C)C(CNC(C2CS(=O)(=O)C2)=O)C1 n1(CC)cnc2c(NC3CCC(SC)C3)[nH]c(=NC3CCCn4ncnc43)nc12 C#Cc1ccc(CC(N2CC(C(N3CC(N(C)C)C3)=O)C(COC)C2)=O)cc1 C1(C(=O)NC2C(NC(=O)CCc3cccnc3Cl)CCCC2)CC2(C1)CC(O)C2 N1(C(C2CC(C)(F)C2)C(c2cccc(O)n2)C)CCC2CN(C3CC3)C2C1 N1(C(c2c(C)c[nH]n2)=O)CC(CNC(C2CCN(C)C2=O)=O)OC(C)(C)C1 N1(C(C(C)=C2CC2)=O)CC(C2CCCN(C(=O)C(CN(C)C)N(C)C)C2)C1 Cc1cc(N)cc(C(N2CCSCC2CCNC(=O)C2=CCS(=O)(=O)C2)=O)c1F C(=O)(CC1=CCCC1)NCC(C)(C)OCC(N1C(CC)CC(O)C1)=O CS(=O)(=O)C1CN(C(C2CC(C#N)C2)=O)CC1NC(=O)Cc1ccco1 c1(C(C)C)nc(NCC2(CO)CC(F)(F)C2)cc(=NC2CCn3nnnc3C2)[nH]1 C1(C(C)C)C(=O)N1.c1(CNC(=O)OC)cccc(CNC(C2CCCO2)=O)c1 C1(SC)CN(C(C2CC(C)CCO2)=O)CC1NC(=O)CN(C1CCS(=O)(=O)C1)C C#CCC(CC(=O)Nc1ccc(CC)nc1C)NC(C1(C#N)CC=CC1)=O N1(C(C2CC(C)(C)C2)=O)CCC2CN(C(c3cc4c(s3)CCCC4)=O)CC2CC1 Cc1ccc(C(C)N(C(c2cc(C#N)ccn2)C(=O)NC2CC2)C)cc1Cl C(=O)(C(C)(C)CSC)NCCC1(NC(C(C)OCCOC)=O)CC1 C1(NC(c2c(COC)cco2)=O)CCN(C(c2oc(Br)cc2C)=O)CC1C c1(C(C)NC(C(c2cccnc2)N(C(C)C)C2CC2)=O)ccccc1 CC(C(=O)N(C)CC1CCCCN1C(C1(F)CCCC1)=O)C(F)F C1(NC(CNS(N)(=O)=O)=O)CCN(C(c2snc(Cl)c2Cl)=O)CC1 c1(N2CCC(OCCNC(c3cc(C(C)C)n[nH]3)=O)C2)ncnc2cccc(F)c12 CC(C)CC(C(N)=O)NC(C1CN(C)CCN1C(C1CCC2(CC1)CC2)=O)=O CC1CCCC1C(=O)NCC(C)(C1CC1)NC(c1nncn1C1CC1)=O CS(=O)(=O)c1ccccc1C(=O)NC1CCC(NC(c2cnns2)=O)CC1 n1(CC)cc(C(=O)NC2CC(CCNC(c3cc(C(C)(C)C)n[nH]3)=O)C2)c(C)n1 C(=O)(C1=CCCOCC1)N1CCC(C)(CCNC(C2(F)CCOC2)=O)CC1 C(=O)(CC(C)CC(=O)NCC(C)NC(=O)Cc1cc[nH]n1)OC c1(O)ccsc1Cl.C1(NC(COCC(C)C)=O)CC(CNC(=O)COC)C1 C1(C)CCCC1CNC(=O)C1CC1.C1(CNC(C2(C(=O)N)CC2)=O)CCCN1SC C1(CC)CCN(C(C2(N(C(=O)C(=Cc3ccccc3)C)C3CC3)CC2)=O)CCO1 C1(C)(C(=O)NCCC2CCCN(C(Cc3cc(C)ns3)=O)C2)CCN(C)C1=O c1(C(N2C(C(C)NC(Cc3c(C)non3)=O)CCC2)=O)cn(C)nc1C(C)C C(C(C)(O)CC(=O)NC(C)CNC(=O)CCN1CCCCC1)OC CC1(C)CC(C(N2CC(CNC(C3CC(O)C3)=O)C3(CC3)C2)=O)C(C)(C)O1 N1(C(CC(CC)C2CCC2)=O)CCOC(C)C1C(=O)NCC1CCN(C(C)=O)C1 c1(CC(=O)NC2CC(CC(=O)NCC(COC)C)C2)cnn(C)c1 c1(OC)ccc(C=CC(=O)N(C2CCOCC2)CCC(=O)O)cc1O C=CCC(C)C(=O)N(C)CC1(NC(=O)C(F)(F)C2(OC)CCC2)CC1 Cc1ccc2[nH]c(C(N3CCC4CC4(NC(=O)C(Cl)=CCl)CC3)=O)cc2c1C n1(CC)ccc2nc(Cl)nc(N(C(C)(C)C)CCc3cccnc3C(F)(F)F)c12 C(=O)(C(O)CCCNC(C12COCC1C2)=O)NC(CCN(C)C)(C)C C=C(C)CCC(=O)NCCCN(C(=O)C(CC=C)c1ccccc1)CC N1(C(C(CC(C)C)NC(c2nc(CC)oc2)=O)=O)CCC2CCC(C2)C1 C1(C(=O)NCC(C)(C)CC2CCCCC2)CCCC1C1CC1.n12cc(nn1)CC2 c1(C(=O)NC2C(CNC(CC=CC)=O)C2)cn(CC(N)=O)nn1 c1(C(N2CCCCC(CNC(=O)CC3CCCOC3)C2)=O)cc2ccnn2cn1 N#Cc1ccc(NC(C2CC23CN(C(c2occc2Br)=O)C3)=O)c2ccccc12 CC1(C)CC(NC(=O)CS(C)(=O)=O)CN(C(c2cc3c(s2)CCC3)=O)C1 C(=O)(CCCC(=O)N1CCC(F)(CNC(C2CC3(CC3)CO2)=O)C1)NC(C)C c1(C(N2CC(O)(CNC(c3c(OC)ncc(F)c3)=O)C2)=O)ccc2occc2n1 c1(-c2cncc(C)c2)cnn2cc(C(=O)NC(c3ccc(Br)cn3)C)cnc12 C=C(C)CCC(=O)NC1CC(CCNC(c2cccnc2CN2CCCC2)=O)C1 c1(NS(CC(C)OC(C)C)(=O)=O)ccc2c(S(N)(=O)=O)cccc2c1 C=CCC(CC=C)C(=O)N1C2CCC1CC(CNC(C1CCCN1C1CC1)=O)C2 C1(C(N(CCCN(C(=O)CNC=O)C)C)=O)CC2(CC2)CO1 C12(C(=O)NCCN(C(=O)CC3C=CCC3)CC)CCC(C)(C1)OC2 C=C1CCC1C(=O)NCCCN(C(=O)C(C)SCCCC)C1CC1 c1(CC23C(CN(C(=O)CC4CC5CCC4C5)C2)CC3)cc(F)cc(F)c1 C12(NC(CC3CN(C)C3)=O)CCCC1N(C(c1cc3cccnc3[nH]1)=O)CCC2 N1(C(=O)NC(CSCC)CC)CC(O)(C(C)C)CC1CO C1(C(=O)NC2CC(CC(N3CC(OC)C(F)C3)=O)C2)CCC2(CCC2)C1 c12ccc3nc(ccc3c1Br)CC2.N1(C(C(=O)OC)=O)CCC(CO)C(C)(C)C1 CCCCCC(C)(C)C(=O)N1CCCC(CNC(C2CCCCCCC2)=O)C1 c1(C(C(=O)NCCC2CC2)N(CCC(=O)OC)C)ccc(C)cc1C N1(C(C2CCCC23CCC3)=O)CCCC2CCNCC12 N1(C(C(=Cc2ccco2)C)=O)CCC2CC2(NC(=O)C=Cc2csc(C)n2)CC1 C1(NC(CCOCC(C)C)=O)CC12CCC(NC(c1cnc[nH]1)=O)CC2 CCCS(=O)(=O)CC(=O)NCC1CC1NC(c1cnc(-c2ccccc2F)s1)=O C1(C(N(CC(COC)O)C)=O)CC=CCN1C(C1CC1CCOC)=O N1(CC(N2CCCC(NC(c3cccc(Cl)c3)=O)C2)=O)CCc2ccccc21 C1(NC(C2CCCS2)=O)CC12CCN(C(=O)CCC1CC1(F)F)C2 C1(NC(C(CNC(C2ON=C(C)C2)=O)(C)C)=O)CCCOC12CCC2 C(=O)(CC(C(F)F)c1ccccc1)N1C(CN)(N)CCC1.c1ccc(F)c(F)c1 C1(NC(CSCCC)=O)CCCCN(C(C2CCC2C(C)(C)C)=O)C1 c1(-n2c(-c3sc(Cl)nc3C)nc(C(C3CC3)COC)n2)cc(F)cc(F)c1 c1(CNC(C2N(C(C(COC(C)=O)C)=O)CCCC2)=O)nc(COC)cc(O)n1 C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)Cc2ccsc2)CC2(CCC2)O1 C1(F)(CNC(C(C)(C)C)=O)CCC(NC(=O)CN2CC(=O)NC2=O)C1 CC1(F)COCCN(C(=NCC=CBr)NCc2ccco2)C1 N1(C(C=CCC)=O)CC(C(=O)NC2CCC(C)(O)CC2)C2(CCC2)C1 CCCC(C(=O)NCC(C1CCC1)NC(=O)Cc1csc2ccccc12)C(C)C CN1CCC(O)C(C2CCCN2C(=O)NCC23CC(CN2CC(F)(F)F)C3)C1 C1(NC(=O)CC2CNC(=O)O2)CC2CC(NC(C3(CF)CC3)=O)CC12 CN1CCC2OCCN(Cc3nc(-c4cnn(C)c4)nn3C3CC3)C2C1 C(=O)(C1=CCCC(C)(C)C1)NC1CN(C(c2n(C)nc([N+](=O)[O-])c2)=O)C1 S(=O)(=O)(c1ccc(F)c(Br)c1)N(CC)Cc1cc(I)c(C)c(I)c1 C1(C(=O)OC)CCN(C(c2sccc2CNC(c2cc(C3CC3)no2)=O)=O)C1 N1(c2cc(C)nc(CO)n2)CCn2ncc(CNC(=O)C(CC(C)C)C(N)=O)c2C1 C1(NC(CC=C(C)C)=O)CCCC12CN(C(C1CCN1C1CCCC1)=O)C2 c1(CC)nc(C)c(C(=O)NC2C=CC(CNC(=O)CCP(C)(C)=O)C2)c(C)n1 C=C(C)c1ccccc1NC(=O)CC1CCCN(C(C2CC(=O)N(C)C2)=O)C1 C1(NC(=O)COCCF)CC2CCC1(NC(c1csc(C3CCCO3)n1)=O)C2 N1(C(C2(CC=C)COC2)=O)CC(NC(C2CCCOC2)=O)CC2(CC2)C1 CN1CCC(NC(=O)COC2CN(C(=O)Cn3ccccc3=O)C2)CC1 c1(N2CCCC(OC)C2)nc2ccc(Cl)cc2c(=NCC2CN(C)CCO2)[nH]1 C1(C(N(C(CC)CC)CC)=O)CC2(CC(NC(=O)CC3CC4CCC3CC4)C2)C1 N1(C(CCC#CC)=O)CCCC(O)(CNC(c2conc2C)=O)C1 C1(COC(C)=O)CCN(C(=O)C(C)CN(C)C)C12CCC2.CCC1C(=O)N1 Cc1n[nH]c(C)c1CC(=O)NC1CC(N(C(=O)C)C)C1.C1(SCC(C)C)(CO)CC1 CCC(CC)(CCNC(=O)CSCc1ccnn1C)NC(c1ccnc(O)c1)=O C(CN=c1[nH]c2c(c(=NC(C)CCC=C(C)C)[nH]1)COCC2)NC(=O)NC CCCCCC(C)(C)C(=O)NCCn1cc(C(N2CCC(=O)N(C)CC2)=O)cn1 c1(C(=O)NCCCN(C(C2C(C)(CC)C2)=O)C(C)C)cc(C(=O)OC)n[nH]1 C1(C(C)C)CCN(C(=O)C2=CCC(NC(=O)CC3CSC3)C2)C1(C)C CCCC(C(=O)N1CCC(N(C(=O)C(C)(C2CCC2)OC)CC2CC2)C1)OC C1(C(=O)NCC2CC(NC(=O)Cc3nc[nH]n3)C2)CCc2ncncc2C1 C1(NC(CC(CC)(F)F)=O)CC2CC(C1)N(C(=O)Cc1ncoc1C)C2 C1(NC(=O)COCC2CCOC2)CCN(C(c2cc(CCO)on2)=O)CC1F c1(OC)cccc(CC(C(=O)O)N)c1.c1(NC(=O)OC(C)(C)C)nc(C)cs1 CS(=O)(=O)C1CC(C(N2CCC(NC(=O)CCc3cc(Cl)no3)C(F)C2)=O)C1 CCCCC(CNC(c1ocnc1C1CCC1)=O)NC(c1ccc(C2CC2)o1)=O N(C1CCc2cccnc21)C(C(N1C(C)C(CO)CCC1)=O)=O C(=O)(C(C(C)(C)C)NC(N)=O)NC12CC(NC(C(CC#C)C)=O)(C1)C2 c1(NC(CC2CCCN(C(C(CCC)CC)=O)CC2)=O)ccc2ncnn2c1 C(C(C(=O)NCC(C1CC1)NC(=O)Cn1nnc(C2CC2)n1)OC)OC S(=O)(=O)(c1ccc(Cl)c(C(=O)NCc2cn(CC3CC3(Cl)Cl)nn2)c1)NC(C)C c1(C(=O)OC)cc(Br)sc1CN1CCC(C(=O)NCC(N)=O)C1 c1(C(N2CCC3(NC(c4cc(CC)oc4C)=O)C(C2)C3)=O)nc(C)c(C)[nH]c1=O C1(CC(=O)NC2CC(C(C)O)C2)CCCN1C(=O)CC1CC(F)(F)C1 N1(C(C(C(CC)C)C)=O)CC2(C1)C(NC(c1ccco1)=O)CCS2(=O)=O C=CC1(CC(=O)N(CCC(O)(CC)CC)C)CN(C(C2CC2C2CCC2)=O)C1 N1(C(C2CCCCS2)=O)CC2CCCN(C(=O)CCc3nnc(C4CC4)o3)C2C1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NC1CC(C(=O)Nc2ccc(I)cc2F)C1 Cc1cccc(C(=O)NC(C2CN(C(=O)CC3CCCC3C)CCO2)C)c1 C1(CC(N2CC(C(=O)OC)C2)=O)N(C(C2CC2(C)C(F)F)=O)CCC1(C)C c1(C(N(CCC)CCNC(C2(C3CC3)CCC2)=O)=O)cnc(Br)c(O)c1 c1(C(=O)NCC2C(NC(C=CC)=O)C2)cc(=O)c2ccc(Cl)cc2o1 c1(C(CN)OC)cn(C(C)C)nc1C.CCCCCCn1nnnc1CC(CC)CC N1(C(C(CCC)OC)=O)C(C)CC2CN(C(c3cccc4oc(=N)[nH]c34)=O)CC12 CC(CCN(C)C)C(=O)NC1CCCC1NC(=O)CNc1ccc(CC#N)cc1 C1(C(N2CC(C3(NC(c4c(CC)n(C)nc4)=O)CC3)C2)=O)CNC(=O)CC1(C)C C12(C3C(CNC(c4cc(C)[nH]c4C)=O)C3)CCCCC1CN(C(=O)C=CC1CC1)C2 N1(C(C(CC)C)=O)CC2(CCC(CNC(c3cnn(C(C)C)c3)=O)O2)C1 n1(CCC)nc(C)cc1C(=O)NCC1(O)CN(C(=O)C(C)Cc2ccco2)C1 N1(C(C(C)(C)C)=O)CC(NC(C2CCC([N+](=O)[O-])CC2)=O)C(C2CC2)C1 Cc1ccc(C(=O)N(CC(C)(C)NC(=O)Cc2ccnn2C)C)c(Cl)c1C c1(N2C3CCC(NC(c4cc(C)sc4C)=O)C(C3)C2)ncnc2ccc(Cl)cc12 C(=O)(CC(F)(F)Cl)NCCN(C(C(c1ccc(CC)s1)=O)=O)C(C)C c1(C(=O)Nc2cccc(C(=O)NCc3cc(C(C)C)no3)c2)cc(O)cc(O)c1 C1(C(N2CCC(NC(C(=O)NCCc3ncc[nH]3)=O)C2)=O)C(F)(F)C12CCC2 N1(C(c2c(C(C)C)scn2)=O)CCCC(CNC(=O)C(C)(C)c2ccns2)C1 c1(CNC(C(C2CCN(Cc3cc(C)[nH]c3C)CC2)C)=O)cc(Cl)nc(Cl)c1 N1(C(C(C(CC)CC)OC)=O)CCCC2(CCCN2C(C2CC3(CC3)CO2)=O)C1 C1(NC(c2c(COC)cco2)=O)CCN(C(=O)CS(=O)(=O)NC2CC2)CCC1CO N12CCC(CC1)C2=O.c1(NC(c2ccc(C(C)=O)[nH]2)=O)cn(C)c(C(N)=O)n1 C1(NC(COCCCC)=O)CC2CN(C(=O)Cc3cnc(C)o3)CC12 N1(C(COCCC)=O)CCC2CN(C(c3ccc(N)cc3Cl)=O)CC12 N1(C(C2C(C=C)CC2)=O)CCCOC(CNC(C2CCCCC2)=O)C1 c1(CC)ccc(Br)cc1C(=O)NCCCN(C(c1cc(C)ns1)=O)CC CCCC1C(=O)N1Cc1ccccc1.C(C)(C(F)F)OC(C1CCCC1)=O CC1OC(=O)NC1C(=O)N(c1ccccc1-n1cc(C(C)O)nn1)C(C)C.CCO N1(C(CS(CC)(=O)=O)=O)CCOC2CCN(C(c3cc(C4CC4)ccn3)=O)CC12 C=C1CC2(C1)C(=O)NC2.C1(OCCSC)CN(C(=O)COC2(C)CCC2)C1 N1(C(CC(C(F)(F)F)OC)=O)CC2(NC(=O)CCN3CCC3)CCCC2(F)C1 c1(C(=O)Nc2ccc(C(N3CC(C#N)OCC3)=O)cn2)c(Br)cc(Br)c(O)c1Br N1(C(c2cccc(C)n2)=O)CCN(C(C2CCC(=O)O2)=O)C(C(C)C)C1 N1(C(=O)CC2CCCO2)CCCC2(CCN(C(C34CC5CC3C4C5)=O)C2)C1 S(=O)(=O)(CC(F)(F)F)N1C(C(=O)Nc2cnc(Br)c(F)c2)CCCC1 C1(NC(c2cccnc2O)=O)CC2CC1N(C(=O)COC1CCOCC1)C2 C1(NC(C(CC#C)C2CC2)=O)CN(C(c2ccnc(CO)c2)=O)CCC12CCC2 CC(CF)CC(=O)NC1CC(COC2(C(=O)Nc3ccccc3)CC2)C1 c1(OC)cc(CC(=O)NCC(C)(C(C)C)NC(=O)CC2CC2)ccn1 CN1CC2(CCN(C(C34CC3CN(C(c3cccc5cncn35)=O)C4)=O)CC2)C1 c1(C(=O)OCC)cc(NCc2c(CCOC)ocn2)ncn1 C(=O)(CCC(O)C(C)(C)C)N1CC(OC)C(NC(=O)C(C)CO)CC1 CCC(F)(F)CC(=O)NCC1CN(C(c2cccc(CO)c2)=O)CC1(C)C c1(CCC(N2CC(CNC(C(CSC)(C)C)=O)OCC2)=O)c(Cl)cncc1Cl c1(OCC(=O)NCC2(NC(=O)CCc3cnn[nH]3)CCOC2)cc(F)cc(Cl)c1 Cc1cc(C)c(C(N2CC(C(O)C(=O)NC34CCN(CC3)CC4)C2)=O)c(C)n1 C=CCC(CNC(=O)CC(F)(F)F)C(=O)NOCCCC1CC1 N1(C(c2cnc(CC)nc2)=O)CC2COCC2(C(=O)NCC2CCCN(C)C2)C1 c1(NC(CCCC(=O)NCC#CCNC(C)=O)=O)cc(Cl)c(C(F)(F)F)c(Cl)c1 CC1=C(C(=O)NCC(C2CCN(C(=O)C3=CCCC3C)CC2)C)CCC1 c1(C(N2CC(N(C(C(C)CC3CCC3)=O)C)C(O)C2)=O)cc2cccnc2cn1 N1(C(C(C(CC)O)C)=O)CC(C2CCCN(C(=O)CCc3ccsc3)C2)C1 N1(C(CCC2(C)CC2)=O)CC(CNC(C2(CC3CC3)CCCO2)=O)C2(CCC2)C1 CCCC(CNC(=O)C(CNC(=O)C=CC1CCC1)CCC)CCO C(=O)(CC(C)C(C)(C)NC(c1nc(C)ccc1F)=O)NCC(C#C)C(C)C c1(C(N2CCN(C(c3ccsn3)=O)C(C3CCC3)C2)=O)cnc(O)c(F)c1 C(CN=C(NCC(F)F)N1CCCC(c2ccccc2)C1)c1[nH]c(=NC)sc1 C1(C(=O)NC(CC(=O)OCC)C)CCCCCN1C(=O)C(CC)n1ccnc1 n1(CC(=O)NC(CC2CN(C(CS(=O)(=O)NC)=O)C2)C)c(C)cc(C)nc1=O C(=O)(C1CCc2ccccc21)NC1CCCCN(C(c2c(C)nncc2)=O)CC1 N1(C(CCSCC(C)C)=O)CC(NC(C2(C)CC2c2ccccc2)=O)C(C)C1 C1(CN(C(C(=O)NCC)=O)C)CCCN(C(C2CC(SC)C2)=O)C1 CC1(C)CCOC(C(N2CC3CCC3(NC(=O)C#CC3(C)CC3)C2)=O)C1 C(C(C(=O)N1CCC(COC)C1)OC)NC(C(OCC)OC)=O c1(CC=C)c(CC2CCC(C3CC3)N2C(=O)N(C)C)nc(Cl)nc1C c1(C(=O)NCC2CN(C(C3CC(CF)C3)=O)CCO2)cccc(C#CC2CC2)c1 CC1(C)CN(C(c2ocnc2C(F)F)=O)CC1NC(=O)CC1CC2CCC(C1)C2 N1(C(C(c2ccnn2C)NC(C(C(C)C)(C)C)=O)=O)CC(O)(C2CCC2)C1 N1(C(c2ncc(C)nc2)=O)CCC(NC(c2nccnc2Cl)=O)C(F)C1 C(C(=O)N(C(C)CN(C)C(C)=O)C)(C(C)(C)C)n1cc(CC(=O)OCC)nn1 C1(C(N(C2(C3CC3)CCC2)C)=O)CC(F)CN1C(C1C2CCC(F)C12)=O N1(C(C(CC)(C)O)=O)CCCC(C)(NC(c2ccc(O)c(C(C)(C)C)c2)=O)C1 c1(NCOC(CCc2c(OC)ccc(F)c2)=O)cc2c(F)cccn2n1 c1(C(=O)NC(CC)CNC(=O)Cc2cocn2)ccc2n[nH]cc2n1 C1(CNC(C2(C=C)CC2)=O)CC2(CCN(C(c3cc(F)cc(Br)c3)=O)CC2)C1 c1(CNC(C(CCC)C)c2nnnn2C2CC2)ccc(C#N)cc1F C1(C(=O)NCCCCC(C)NC(=O)CC2COCCN2C)Cc2ccccc2C1 N1(C(C(Cc2ccsc2)NC=O)=O)CCOCC(CNc2ncc(Cl)cn2)C1 CC1=NN(C)C(=O)C1CC(=O)NCC1(CNC(c2cccc(O)c2Cl)=O)CCC1 C(C(C)(C)CC(C)O)NC(COCCNC(C1CC=C(C)CC1)=O)=O c1(C(=O)OC)nc(N2CC3CC3(CNCC3(c4ccccc4)CC3)C2)ncc1F C1(C(=O)NCC(C)CNC(c2cn(C(C)(C)C)nn2)=O)CCCCC1(F)F N1(C(C(=O)N(C)C)=O)CCC2C(CCCN2Cc2coc(-c3ccccc3)c2)C1 CC1CCCC1(C(=O)NCCC1CC(F)(F)C1)NC(c1cc(CC2CC2)on1)=O c1(OCC)ccnc(NC(C)CNC(=O)CNC(c2cccc(C)c2)=O)n1 C1(NC(=O)CCc2cnn[nH]2)CC(O)CN(C(=O)CN2CSCC2=O)C1 c1(C(=O)NCC23CC(CNC(CC(C=C)(C)C)=O)(OC2)C3)ccc(F)c(O)c1F C1(C(N2CC(CCNC(C(C)(C3CC3)OC)=O)C2)=O)CNC(=O)CC12CCC2 N12CCC(C3CC3)(C1)CN(CC)C(CC)C2=O.C1(C(=O)NC)(C(=O)N(C)C)CC1 C12(C(N3CCC(CC=C)(NC(C4(CO)CC4)=O)CC3)=O)OCCCC1C2(F)F N1(C(c2cc(-c3ccccc3Cl)no2)=O)CC2C(CNC(C3(CF)CC3)=O)C2C1 c1(OCC)nc(C(=O)NCC(CC)NC(C2CCCN2CC)=O)ns1 CC(C)C(CNC(c1cccc(C(C)S(N)(=O)=O)c1)=O)C(C)C c1(C(=O)NCC(CN(C(=O)Cc2ccnn2C(F)F)C)O)cnn(CCO)c1 N1(C(COCC#C)=O)CCC(C)C(N(C)C(c2cc(C(=O)OC)no2)=O)C1 c1(NCc2c(C)ccnc2)cc(Br)ccc1S(=O)(=O)NCCN=c1cncc[nH]1 c1(C(N2CCC(O)(C(C)CNC(c3ccoc3C3CC3)=O)C2)=O)cc(F)cc(F)c1 c1(CC)cc2c(CC(=O)NC(C)C(C)NC(=O)C(C)COC)csc2s1 N1(CC)CCCCC1C(=O)NC1CN(C(=O)C(F)=C(C)C)CC1OC N1(C(C(C(C)C)c2cnc(C)s2)=O)CCCC(CNC(=O)C=C2CCC2)C1C C1(c2cn(C)nc2)CC1N=c1[nH]c(=NC2CCSCC2)[nH]c2ncn(C)c12 C1(c2n(CCSC)nnn2)(NC2(C)CC=CCC2)COC2(CCC2)C1 C1(CC(=O)N(C2CCN(C(=O)Cc3cn[nH]c3)C2)CC)C(=O)N(C)N=C1C c1(OC)ccc([N+](=O)[O-])c(NC(=O)Nc2ccsc2OCC(F)(F)F)n1 C1(NC(c2ccc(C#C)cc2)=O)CCN(C(c2nncn2CC)=O)CC12CCC2 O=C(CCC(F)F)NN1CCCC1C(=O)NC1CCC(O)CC1 C1(C(=O)NCC2CCC(NC(=O)COC3CCOC3)C2)CC12CCS(=O)(=O)CC2 C(C(C)C(F)C(=O)NCCN1CCC2CC12)NC(Cc1c(C)ccnc1)=O C(CCCCC(=O)NCC1CC1)=CC.c1(C(N2CCC2)=O)csc(-c2ccsc2)n1 C1(C(C)NC(=O)NCc2cnns2)CCCCO1 C(=O)(C1=CCCCC1C)NC(c1occ(C(=O)NCC(C(C)O)(C)C)n1)C CC1=C(C(=O)N2CC3CCCC3C2C(=O)NC(C)C(=O)NC(C)C)COCC1 n1(C(c2c(C)cccc2)c2nnnn2C)c(=O)oc2ccccc12 c1(C(=O)OC)cc2[nH]c(C(N3CC4CC(NC(=O)CCS(C)=O)C4C3)=O)cc2s1 C12(C(=O)NC3(C)CCCN(C(=O)CC#N)C3)CC3CC(C(=O)N1)C2C3 C(=O)(C1=NOC(C)C1)NC1(C)CN(C(c2n(CC)ccn2)=O)C1 C1(F)(CNC(CCSC)=O)CCC(CNC(=O)C(C2CCCCCC2)O)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCC(O)CNC(=O)Cc2ccoc2C)c1Cl N1(C(Cn2cc(CC[SH](C3CC(C(=O)O)C3)C)nn2)=O)CCOCC1C C(=O)(C(O)C(F)F)Nc1cn(C2CCOC2)cn1.c1(N2C(=O)C2)ccc(O)nc1 c1(N2CCC(NC(c3nncc(OC)c3)=O)C(F)C2)ncc2c(n1)COC2 C(CO)(CCCCNC(=O)C(O)C(F)F)NC(c1c[nH]nc1[N+](=O)[O-])=O CS(=O)(=O)c1cc(C(N2CCC(NC(c3ccc(=O)oc3)=O)C(CO)C2)=O)co1 N1(C(c2occ(C(C)=O)c2)=O)CCC(CO)(NC(=O)CC(C)n2ccc(C)n2)C1 c1(C(=O)NC(c2ccc(Cl)nc2)C(F)(F)F)cc2ncnc(O)c2cc1Cl c1(CC)nn(C)cc1C(=O)NCCCC1CCCCN1C(C1CC(=O)N(C)C1)=O C12(NC(CC)=O)CCN(C(=O)CCc3ccc(OC)nc3)CC1C2 c1c(COCCN=c2nc(C3CCOCC3)[nH]s2)sc2c1CCCC2 N1(C(C(C)(C)Oc2ccc(Cl)cn2)=O)CCC(C)(c2ccc(F)cc2)CC1 c1(C(C)C)cc(C(=O)NCC(CO)NC(=O)C(F)n2cccn2)ccc1F c1(C(=O)NC2(C)CCN(C(C3(C)CCC3)=O)C2)ccc(Br)c(O)n1 C1(C#CC(=O)NCC2CN(C(=O)CC3CCCCC3)CCC2C)(CC)COC1 C12(NC(c3ccnn3CCF)=O)CCN(C(=O)CSCc3ncc[nH]3)CC1C2 Cc1ccc2c(c1)SC(C(=O)NC1CC(C)CN(C(=O)C=C3CCCCC3)C1)C2 C(=O)(CCC(=O)N1CCC(O)CC1)NCCC(C)N(C)C(C1CCO1)=O c1(C(N2C3CC(CNC(C4N(CC)CC4)=O)C(C3)C2)=O)cnn2c1OCCC2 c1(C(=O)NC2(C(N(C(C)CC(N)=O)C)=O)CC2C)ccc(=N)[nH]n1 N1(C(c2cn(C)c(=O)cc2)=O)CCN(C(=O)CCSC(F)(F)F)CC(C)(C)C1 C(N=c1cc(C)n(CCOC)[nH]1)c1c(CC)nn(C)c1 CC1CC(NC(C2CCCS2)=O)CCN1C(=O)CSC(F)(F)F C(CCC(=O)N1CC(CO)C(C(C)C)C1)(C(C)C)NC(C1C(CC)N(C)CC1)=O C1(N(C(c2ccc(CC)s2)=O)C)CCN(C(=O)C(O)CC)CC1 C1(NC(CCNC(CC2CC(C)C2)=O)=O)CN(C(=O)CN(C)C)CC1C c1(OCC)ccc(NC(=O)CN2CC3(CCCC3c3nn[nH]n3)C2)c(Cl)c1OC c1(CN(CCCCCC)C(=O)C(N2CCC(NS(C)(=O)=O)C2)=O)cccc(Cl)c1 C1(NC(Cc2ccc(OCC)cn2)=O)CN(C(c2csnn2)=O)CC2CC12 C(=O)(CC(C)C(F)(F)F)N(C(C)C(=O)NCC=CCCC)CC=C c1(C(=O)NC2CC(NC(=O)Cc3ccccc3O)C2)ccc2c(c1)S(=O)(=O)NC2 C1(C(=O)NCC(CC(C)C)CO)CC(N=[N+]=[N-])CN1C(=O)CCC1CCC(=O)C1 c1(C(C)=O)ccc(C(N2CCC(O)(CNC(=O)C=Cc3cnc(C)s3)C2)=O)nn1 C1(CC(=O)N(C2CN(C(=O)CCC3CC3(Cl)Cl)C2)C)CSCCS1 N1(C(c2cccc(CNC(c3cn(CC)nc3C)=O)n2)=O)CC2CC(C)C2C1 C#CCCCC(C)C(=O)NCC1CN(C(C2CCCN2C)=O)C1 C(=O)(CC(C)C(F)(F)F)NC(CC(N(C(c1cc(F)ccc1O)C)C)=O)C C1(CC)CN(C(c2cccc(C(C)C)c2)=O)CCN1C(=O)C=C1CCN(C)CC1 CC(CO)CCN=c1[nH]c(N2CCC3(CC2)CN(C)C3)nc2c1CCC2 C1(CCNC(CCN(C(CC2CC(=C)C2)=O)CCO)=O)CCC(C)(C)O1 c1(NC(C(N2CC(c3n(C)ncc3)(O)C2)=O)=O)cc2cc(Br)ccc2s1 C(=O)(CCCCCO)NCC(C)CN(C(=O)C1=COCC1)C c1(OC)ncccc1NCc1ccccc1SCc1ncccn1 c1(C(N2C3(C(=O)NCc4c(C)nccn4)CC(C2)C3)=O)cc2ccccn2c1 Cc1sc(Cl)c(C(N2CCCCC(CNC(=O)C=CC3CCOC3)C2)=O)c1C C1(C(=O)NC2(CO)CN(c3ncnc(OC)n3)C2)CC2CCCCN2C1 CCC(C)(C)C(=O)C(=O)N1CCC(CC(N2CC(OC)C(O)C2)=O)C1(C)C CN1CCN(C(=O)CCc2nc[nH]n2)CC1C(=O)Nc1cccnc1 CCC(C)(C)C(O)C(=O)NCCN(C(=O)C=CC(C)CC)C.OC c1(CC(=O)NC2CCN(C(C(C(C)C)SCC)=O)C23CC3)cccc([N+](=O)[O-])c1 C1(OCC(=O)NCCCN(C(C(C)=CC)=O)C2CC2)CCCCC1C CC(Cl)(Cl)C(=O)N1CCC(CCC(=O)N(C2CC2)Cc2cccs2)C1 c1(N2CCC(C(N3CCN(C(C45CC(CO)(C4)C5)=O)CC3)=O)C2)ccccc1Cl N1(C(C2C(C(=O)OCC)C2)=O)CCC2(CC1)CC(C)N(C(=O)COC(F)(F)F)C2 CCC(C)CC(=O)C(=O)NCCn1ccc(C(=O)NCCOC2CC2)c1 c1(C(N(CCN(C(C(CCOC)C)=O)C)C)=O)cncc2c1CCCC2 CCC(CC(=O)NC1CC(OC)C1)N(C)C(c1cccc(O)c1)=O C#CC1(O)CCN(C(=O)CC2CCC(NC(=O)CCCCC(=O)OC)C2)CC1 C1(O)(c2cn(Cc3cccc(C)c3)nn2)CCN(C(C2CCC(=O)N2)=O)CC1 C1(CNC(=O)C(O)Cn2cncn2)CC(O)CN1C(c1ccc(Cl)o1)=O C(CN=c1nc(C)cc(C)[nH]1)C1N(C(C(c2ccc(C)cc2)C)=O)CCCC1C c1(C(=O)NCC(CN(C)C(C2(C)CCCO2)=O)O)ccc(N)cc1O C1(N=[N+]=[N-])(C(=O)NCC(C(CC)C)CO)CCN(C(=O)CN2CCCC2=O)C1 Cc1ncncc1C(=O)NCC1CC1NC(=O)Cc1ccsc1C CON=CC(=O)NCC(C)(Cn1cccn1)NC(C1CC(=O)C1n1cccn1)=O c1(C(N(C(C)CNC(C2CC=CC2)=O)C)=O)cc(C(F)(F)F)ccc1N N1(C(C(CCSC)NC(C2CCC(C)(C)CC2)=O)=O)CCC(C)(C2CC2)C1 C(CCCS(C)=O)NC(CCN(C(C1CC1F)=O)CC)=O CCCCC(CC(=O)NCc1noc(C(N)=O)n1)NC(C1(C)SCCCS1)=O C1(CC(N2CC(CCNC(C(C)OCC)=O)(OC)C2)=O)CCCCC1C(F)(F)F c1(C(N2CCN(C(C)C(N3CCCC(O)C3)=O)CC2C)=O)cnn2ccccc12 c1(CC(=O)NC2CCCC(CNC(CC3(C)CC3)=O)C2)cc(F)cc(F)c1 C1(C(=O)NC2C(CC)N(C(=O)CC(F)F)CC2)CC2COCC2C1 n1(CC(N2C(C3(O)CN(C(CC4CC(OC)C4)=O)C3)CCC2)=O)cnccc1=O N1(C(CCC(=O)NC)=O)CC(C)C(NC(c2cnn(C)n2)=O)C(C)C1 S1(=O)(=O)c2ccc(cc2)NCC(=O)N1.c1(C(=O)OC)ccc(C2CC2)s1 C1(C(C)(C)C)(CNC(=O)CO)CCN(C(C2CCCCC2c2nc[nH]n2)=O)C1 C12CC(C1)CC(=O)N2.C1(F)(C(=O)NC2(CCCC)CC2)CC1C C1(CNC(C(n2cc(-c3ccnn3CC(F)F)nn2)C)=O)CCCCC1(F)F C1(C(=O)NC2C(NC(CCN(CCC)C)=O)CCOC2)CCCCCS1(=O)=O C(=O)(C1=CC(C)CC1)NCC1(NC(Cn2c(C)c(Cl)cn2)=O)CCC1 C(=O)(CCCCC(N)=O)NC(C(C(C)C)NC(CCC)=O)C.C1(=O)CN1 CN1CCC(NC(=O)CC=CCNC(=O)C(F)(F)C2CC2)C1(C)C C1(C(=O)NCC=CCSC)(COC)CCN(C(C2(C)CCOC2)=O)C1 CC1(C(N2CCC(C)(NC(=O)COc3cccnc3)C2)=O)CC(C(F)(F)F)=NO1 CN1N=C(CC(=O)NC2COCC2NC(c2ccn3ccccc23)=O)CC1=O CC1COCC(C(N2CCC(C(N3CCC(O)(CO)C3)=O)(CF)C2)=O)O1 N1(C(CCCOCC)=O)CC(C)CN(C(c2ccc(C)c(F)n2)=O)CC1C C1(NC(=O)Cc2cc(O)ccc2Br)CCc2nc[nH]c2C1 c1(CCN(C)C)cccc(C(=O)N(CC(O)CNC(C2(C)CCC23CC3)=O)C)c1 C1(C)(CC)CCC(C(=O)NCC(C2CCCN2C(=O)CSS(C)(=O)=O)(C)C)O1 c1(CN2CCC(N(C(c3nn(C)cc3Cl)=O)CC)C2)c(O)nnc(C)c1C C1(C(=O)NCCCC(C=C)(C)C)CN(C(=O)CC(C)C(F)(F)F)CC12CCC2 Cc1nnc2n1CC(C(=O)NCC(n1cc(C3CCC(CO)CC3)nn1)C)C2 Cc1ccc(CC(N2CCC(C)(C(=O)Nc3cccc(F)c3C)C2)=O)c(C)c1 CN1CCCC(C(=O)NC2CC2NC(c2ccc(Cn3ccnc3)cc2)=O)C1 N1(C(CCCCC)C)CCC2(CC1)CC2(C)C(=O)NC1CCOC(C)C1 C1(CCC(=O)NCCCN(C(C2(CCF)CCC2)=O)CC)CCCN(C)C1 C1(NC(C2(F)CCN(C(=O)CCc3cocn3)C2)=O)CCCCNC1=O c1(C(=O)NC(C(=O)NCC2(C)CCN(C)C2)c2ccoc2)ccc(F)c(O)c1 N1(C(N(c2cnccc2C)CC)=O)CC2(CCCCC2)c2ccccc21 c1(C(N2C(C(=O)NC3(C(C)C)CC3)CC=CC2)=O)c[nH]c2ncccc12 CC1(C)CN(C(c2cccnc2)=O)CC2(CN(C(C3CC4(CCCC4)C3)=O)C2)O1 c1(OC)cc(Cl)ccc1C(=O)NCC1CN(CCCCCF)CCO1 c1(C(=O)NCC2(F)CC(NC(C(F)=CCC)=O)C2)cc(O)nc(SC(C)C)n1 c1(NC(C(C(C)NC(c2c(NC)scn2)=O)C)=O)ccc(C)cc1C C1(C(NOCCCOC)=O)CCC(CO)O1.C12(CC1)C(=O)N2 Cc1ccc(C(N2CC=CCC2C(=O)NCC(C)(F)C(C)(C)F)=O)nc1O CN1CC=C(C(=O)NCCC2CN(C(C3CC(=O)N(C)C3)=O)CCCO2)C1 c1(CNC(C2CCN(C(c3ccc(I)cc3)=O)C2)=O)cncc(NCC(F)(F)F)c1 c1(C(=O)NC2C3(CN(C(C(C)(Cl)Cl)=O)C3)CC2)ccc(F)c2ccccc12 C1(=O)N2CCC(O2)NC(=O)C2C1CCC2.C1(COC)CCCOCC1 C1(CC)CNC(=O)CN1C(=O)C(CNC(C1CC(=O)N(OC)C1)=O)C(C)C c1(C(=O)NC2CN(C(C3CC(OCC)C3)=O)CC2C)cnc2c(c1)CCC2 c1(C(=O)NC(CNC(C(CCSC)OC)=O)C2CC2)coc2c1NC(=O)CCC2 n1(CC(=O)NCC2(F)CN(C(C3CCC3(F)F)=O)C2)cc(Br)ccc1=O c1(NC(=O)NC2C(CCC)C2)ccc(C(C)(C)C)cc1[N+](=O)[O-] c1(N2CCC(NC(C(C)(C)F)=O)C2)ncnc2c1CCO2 N1(C(C=CC(C)C)=O)CCC(C2CCN(C(c3cnc(C(F)F)cn3)=O)C2)CC1 N1(C(C2C3(CCN(C(Cc4n(C)ccc4)=O)C3)C2)=O)CC2(CCCCC2)C1 c1(NCC2(OCC)CCC2)ccc(S(=O)(=O)N2CCN(S(C)(=O)=O)CC2)cc1Br N1(C(=O)Nc2ncc(C(F)(F)F)s2)CCC(c2cccs2)CC1 c1(N(C(C)=O)C)ccc(NC(CN(C)C(c2ccc(C(F)(F)F)cc2)=O)=O)cc1 N1(C(c2cccn(C3CCC3)c2=O)=O)CCN(C(C2CC=CCO2)=O)C(C2CC2)C1 c1(CC)ccc(C(=O)N(C)CC2CC(F)CN2C(c2csc(COC)c2)=O)cc1 c1(C(N(CCNC(CCc2c(C)ncs2)=O)C(C)C)=O)cn(C)c(=O)cn1 Cc1cc(C#N)ccc1C(=O)NOCC(=O)NC(c1ccc(F)cc1F)=O C=CCCCCCC(=O)NC1C2CCN(C(c3ccc4c(c3)OCO4)=O)C12 C1(NC(CCC#C)=O)(CO)CCN(C(c2ccc(C)[nH]2)=O)CC1 CC(C)(C)CCCC(=O)NC1CCCCC12CCC2 c1(CN(C(=O)C(N2COCC2(C)C)=O)CCCC)ccc(F)cc1 c1(CC)cccc(-c2cn(CCCCC(=O)N(CC(F)(F)F)C)nn2)c1.C1CO1 c1(C(=O)NCC2C(NC(CCOCCC)=O)CC2)nc(C2CC2)cs1 C(CCC(O)CO)NC(=O)C(=O)N1CC(=CC2CCCO2)C1 Cc1cncc(C(N2CCCCC2C2CCN(C(C3(C)COC3)=O)C2)=O)n1 C(C)(CCCC(=O)N1CCOC(C(C)C)C1)NC(C1C(=C)C1)=O C1(NC(c2c(CC)scn2)=O)CN(C(c2ccc(C#N)cn2)=O)CCC1CO c1(CC(=O)NC(CN(C(C=C(CC)CC)=O)C)(CO)CO)ccc(C)cc1C C12(NC(C3(C(=O)OC)CC3)=O)CC1CN(C(c1occc1Cl)=O)C2 n1(CC)c(N2CCN(C3CCN(CC(F)F)C3)CC2)nnc1-c1ccc(O)nc1 C(C(CC(=O)NCC1(O)CCCOC1)C1CCC1)NC(C1C(C)=CCS1)=O c1(C(c2nnnn2CCCF)NCC(COC)C)cccc(OC)c1C CC1CCc2nc(C(N3CCCCC(NC(=O)Cc4cncn4C)C3)=O)cn2C1 Cc1nn(C)c(C)c1OCC(=O)NCC(O)CN(C(=O)CC1OCCO1)C N1(C(CN(C(COCCCC#C)=O)CC#C)=O)CC(C)c2ncccc21 C1(O)(C(=O)NC(C=C)C)CCN(C(C2(c3cccs3)CCCCC2)=O)CC1 Cc1ccc(CCC(=O)N(CCCn2cc(COC3CCOC3)nn2)C2CC2)s1 C1(NC(c2nccc(CC)c2)=O)CN(C(C2CC(=O)NC2(C)C)=O)CC1(C)C c1(NC(C(CC=C)NC(=O)CC(C)(C)COC(C)=O)=O)cc(C)ccc1Cl c1(OCC)cccc(NC(C)C(N2CC(c3ccccc3Cl)(F)C2)=O)c1 Cc1cccc(CS(N2CC(c3ccccc3)(C(N3CCSCC3)=O)C2)(=O)=O)c1 C1(NC(CC(CC)(F)F)=O)CC2CCC(C1)N2C(C1CC(C)OC(C)C1)=O c1(OC)cc(C(=O)NCC2CC3CCC2N3c2cc(C)nc(Cl)n2)ccc1C#N C(CCCC(=O)NCCCN(CCCNC(=O)C(C)COC)C)CC.OCC N1(C(C(F)OC)=O)CCC2(CCCN2c2ccc(C#N)c(C#N)n2)CC1 C1(CNC(c2cnoc2)=O)CC2(CCOCC2)CN1C(c1ccc(O)c(O)c1)=O N1(C(C2(C)N(C)CCC2)=O)CCCC2CN(C(=O)C=C3CCCC3)CCC12 C(=O)(CCCCCC(C)O)NCC(=C)CCNC(C1CC1C(F)(F)F)=O c1(COCC(=O)NCC(CNC(c2c[nH]nc2F)=O)OC)nnc(S)n1C C(CCCCCN(C)C(c1n[nH]c(C)c1C)=O)NC(COCCCC)=O N1(Cc2nnc(C(C)C)o2)CCCC(CO)(NC(=O)CC2CCC(C(N)=O)O2)C1 c1(OC)ccncc1-n1cc(COC2CCN(C(=O)COC3COC3)C2)nn1 C1(CCOC)CN(C(=O)CC(Cl)Cl)CCN1C(=O)CCCSC(C)(C)C c1(OC)ccc(Cl)c(C(=O)NCCC2CN(C(=O)C3=CCC3)CC(C)O2)n1 C(=O)(C(C)C(F)(F)C(F)F)NC(C(=O)NCC(CC=C)CC(C)C)COC c1(C(c2nnnn2CC2CCOCC2)NC(C(=O)NC)C)nc(C)c(C)nc1C O=C(N=c1ccn(Cc2ccccc2)[nH]1)C1CC1CCc1cccs1 c1(C(=O)NC(CCCC)C(=O)N2CCCCC(C)C2)cc2ccccn2n1 N1(C(CN(CCC)C)=O)CC(N(C)C(c2cc(Cl)nnc2O)=O)C2(CC2)C1 CC(CN(C)C)CCC(=O)NCC1(C)CCN(C(=O)C=Cc2ccsc2)C1 c1(CC)ccc2cccc(NC(N3CCC(OC)C3C)=O)c2c1 c1(CNC(C2CCC3(CC3)N2Cc2c(C)ocn2)=O)cccc(C#N)c1C n1(C(C23C4(CC42)OCC3)(CC)COC)nc2ccccn2c1=O c1(OC)cc(C)sc1C(=O)NCC(C(C)C)NC(=O)C=Cc1nc(C)cs1 C(=O)(CCN(C(=O)CSC1CC1)C1CC1)N(CC(C)OC)C C1(NC(C2(C)N(C(=O)OC(C)(C)C)CC2)=O)CCOCC1CNC(=O)CNC=O C1(NC(c2cccs2)=O)CC2CC1CN(C(c1cccc(OC(F)(F)F)n1)=O)C2 c1(C(=O)NC2C(C)CN(C(=O)CC3CCSCC3)C2)ccn2cccc2c1 CC1CC(C(=O)N(CCCNC(=O)C2=CCCS2)CCO)CC(C)C1 C1(CNC(CCNC(N)=O)=O)CN(C(=O)CC(c2ccc(Cl)cc2)O)CCO1 C1(C(=O)NCC2(NC(c3scc(C(C)(F)F)n3)=O)CCOC2)CCn2ncnc2C1 C1(C)CC(=O)N1.C(COC)(C(=O)OC)N.CCCC(=O)NCC1CC1 CCCCCC(O)C(=O)NC1CCN(CCCC(C)=CC)C1 c1(C(=O)NC(C)CN(c2ncnc(C#N)c2F)C)cnc2[nH]c(O)nc2c1 c1(CCNC(C2N(C(c3ccc(C)n3C)=O)CCC2C)=O)cn2c(n1)CCCC2 C1(N(CCCC)C(C2CC2F)=O)CCN(C(C2CCCN2C)=O)CC1 Cc1cn2cc(C(=O)C(=O)NCCOc3ccccc3[N+](=O)[O-])nc2s1 C12(NC(=O)CCc3ccc(O)nc3)CCN(C(C3CCC=CCC3)=O)CC1C2 Cc1cc(NC(=O)NC(C(C)NCc2cccc(N(C)C)c2)=O)cc(O)c1 C(CCCS(C)=O)NC(C(COC)NC(C(COC)N(C)C)=O)=O.N(C)C N1(C(Cn2ccc(=O)n(C)c2=O)=O)CCC2CN(C(=O)CC3CCC3)C2C1 c1(CNC(=O)CO)cccc(C#N)c1.C(=O)(CCCCC(COC)=O)NCC(CO)O N1(C(Cn2nc(C)oc2=O)=O)CCC(C(=O)NCC(Cl)Cl)CC1C Cc1ccc(C(=O)NC2CC3(C2)CC3C(=O)NCCCC(C)(C)CO)c(O)c1 c1(CC)cc(C(=O)NCC(C(C)(C)C)NC(C2CC3CCC3C2)=O)cc(N)c1 Cc1cc(C(=O)NCC(C)N(C(=O)Cc2c(C)noc2C)C)ncc1N c1(C(C)NC(c2n(CC)nnn2)c2ccn(CCOC)n2)ccc(Br)c(Cl)c1 CC1CS(=O)CCN1C(C1CC2CCC1N2C(c1ncccc1Cl)=O)=O C1(C)(C(=O)NC(CC)CNC(c2cccc(CN3CCSCC3)c2)=O)CC2CCC1O2 C1(C(=O)NC2(C)CC(NC(=O)Cc3cnc[nH]3)C2)COCCN1C=O N1(C(c2c(CC)n(-c3ccccc3)nc2)=O)CCC(NC(=O)CCOC)C1(C)C C1(C(N2C3CC(CC(NC(C(C)(C)F)=O)C3)C2)=O)CCCCC12OCCO2 Cn1ncc2cc(C(=O)NCCCN3CCN(c4ncnc(Cl)c4F)CC3)sc12 N#Cc1ncccc1S(=O)(=O)N(c1ccc(Cl)cc1)CC1CSC1 c1(CNC(=O)CCOC2CCCC2)cn(CCCO)nn1.C12CC(CO1)C2 N1(CCNC(c2nccc(C(F)(F)F)n2)=O)Cc2ccc(Br)cc2C1=O n1(CC(=O)NCCCC(C)NC(c2cccc(F)c2O)=O)cc(S(C)(=O)=O)cn1 C(=O)(C#CC1CCCCC1)N(C)CC1CCC(C(=O)O)CC1 C1(C(CNC(C(C)SCCCC)=O)O)CCN(C(c2cncn2C)=O)CC1 N1(C(C(C=CCCC)O)=O)CC(CNC(=O)CCc2cn[nH]c2)OC2(CCC2)C1 CCC(O)CCN=c1cc(C)c(S(=O)(=O)NCC2CC(O)CCO2)c[nH]1 N1(C(c2sc(C)c(O)n2)=O)CCC(NC(=O)Cc2cccnc2Cl)C(C)C1 c1(CN2CCC(OC)(CN(C)C)CC2)cnc2ccccc2c1 c1(C(=O)NC(C(=O)NCC(C)OCC=C)Cn2cncn2)cc[nH]c(=NC)c1 N1(C(C2CCC(=C)CC2)=O)CCC(NC(C2CCCCNC2=O)=O)C12CCC2 N1(C(=O)CCC2CCOC2)CCC2C(C(N3CCCC4(C3)N=N4)=O)C2C1 CCC(C)CC(C(=O)O)N(CC(=O)Nc1ccccc1)Cc1ccccc1OC c1(C(N(CC(C)N(C(=O)C(F)C(F)(F)F)C)C)=O)cccc(F)c1F C(=O)(C1=COc2ccccc2O1)NC1CC(CNC(=O)CCC[N+](=O)[O-])C1 C1(CCC)CCCN(C(c2cnn3c2C3(C)OC)=O)C1.N1(CC(=O)OC)CC2CC2C1 O=S(=O)(c1cc(Br)c(Cl)s1)N1CCC(O)CC12CC2 n1(C(c2ccc(F)cc2)C(C)C)c(N)c(C(=O)CNC(=S)N(C)C)c(=O)n(C)c1=O c1(OC)cc2ccccc2c(C(N2CCN(C(c3ccccn3)=O)CC2C)=O)n1 N1(C(C2C(C)OC(C)C2C)=O)CC2CC1(c1cn(CC(O)C(F)(F)F)nn1)C(=O)N2 N1(C(c2c(C)cc[nH]2)=O)CCC(F)(CNC(C2CC2(c2ccccc2)C)=O)C1 c1(C(N2CCCC(c3nccs3)C2)C(=O)NCC)cccc2cnn(C)c12 c1(NC(C2C(C(=O)NCC(c3ccc(C)cc3)O)C2)=O)nc2ccccc2s1 C1(CNC(=O)CCCc2cc[nH]n2)COCCN(C(c2cnco2)=O)C1 CCC(C)CC(=O)NCC1(OC)CN(C(c2ccccc2SCC(F)(F)F)=O)C1 N1(C(c2cccc(NC)n2)=O)CC2CCCC(C1)N2C(C1CC(C)(F)C1)=O C1(C(C)NC(=O)CCCC2CCOCC2)CCCN(C(=O)C(O)CC2CC2)C1 c1(SC)ncc(N)c(C(=O)NCC2CCC(C)C2)n1 C(CCN=c1[nH]c(=NCCC2CCCC(C)C2)[nH]c2c1CCCC2)OC C1(C)(CCCCC#N)C(CCC)N1CC1CC1.c1(CO)cc[nH]n1 N1(C(CC(CC)C)=O)CCC2(CC2C(N2CC3CC3C2C#N)=O)C1 c1(CC(=O)NC2CCC(NC(c3ccns3)=O)C2)ccc(F)c(Br)c1 c1(C(=O)NCC(CNC(C=Cc2c(C)cccn2)=O)F)c(F)cccc1[N+](=O)[O-] c1(C(N(CC(C)(C)NC(C)C(=O)NC(C)(C)C)C)=O)cc(C2CC2)ns1 N1(C(C(CC)Oc2ccc(C)cc2C)=O)CCC2(CC1)CNCC2C(=O)O c1(C(=O)NCCCCCn2cc(C(C)(C)OCC)nn2)cc2ccccc2nn1 c1(C(N(CC(=O)NC(C)(C)CC2CCC2)CC)=O)cscc1OC C1(CC(=O)N(C)CCNC(CCOCC#C)=O)CCCCO1 N1(C(CC(CC=C)c2ccccc2)=O)CC(C(=O)NC2CC2)C(C2CC2)C1 c1(C(=O)NC(CC)CNC(C2CN(C)C(=O)N2)=O)cccc(C#CC2CC2)c1 CC(CCCNC(=O)CCC1CCOC1)NC(=O)C(C)Sc1ccccc1 c1(C(N2CCC(C)C(NC(c3ncccc3CO)=O)C2)=O)ccc(Cl)c(C#N)n1 CC(C)CC(F)(F)C(=O)NC1CCCC(NC(c2ccc(F)c(F)c2)=O)CC1 c1(OC)cc(OC)c(C(N2CC(C)C(N)C2)=O)cn1 CC(C)CS(=O)(=O)CC(=O)N1CCN(C(C2CCC(=O)N2C)=O)C2CCC12 C1(NC(CC(C=C)(C)C)=O)CN(C(c2ncccc2SCC)=O)C2(CCCC2)C1 C1(C(=O)NC(=O)OC(C)(C)C)CN(Cc2cc(O)nc(C3CC3)n2)CCN1C(N)=O N1(C(C2N(CCC)CCC2)=O)CC(C)(C)CC1C(=O)N(C)C1CC1 c1(C(=O)NC(CNC(C2C(CCC)C2)=O)CCOC)cc(Cl)c2c(c1)OCCO2 c1(C(=O)NCCN(CCC)C(C2CNC(=O)C2)=O)n[nH]c2ccc(OC)nc12 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1CC2N(C(COCC)=O)C(CC2)C1 N1(C(C2C(C=CC)CN(C(=O)CC(C)C)C2)=O)CCCC2(CC(O)C2)C1 C1(C(=O)NC2CCN(C(CC(COC)C)=O)CC2)CCn2nnnc2C1 c1(C(=O)NCC(C)(CC)NC(CCCCC)=O)cc2ccccc2c(O)n1 c1(OC)cc(CNC(c2ccccc2-c2cccnc2)=O)cc(OC)c1Br C1(c2c(COC(C3C(C(C)C)OCC3)=O)cnn2C)CC2(CCO1)CC2 C1(C)(C(N2CC(CNC(c3nc(CC(C)C)sc3)=O)C(C)C2)=O)CCC(O)CC1 C1(C(C)C)CN(C(=O)CN(C)CCN(C)C)CCCN1C(=O)Cc1ccnn1C c1(C(N2C(C(=O)NC3CC(C(=O)OC)C3)CCC2)=O)ccc(CNC(C)=O)cc1 CC(C)C(C)C(=O)NC1CCCC1CNC(=O)CCOCCOCCCO N1(C(C2C(C)=C2)=O)CC(NC(=O)CS(C)(=O)=O)C(C)C1 C1(C(N2CC(SC)C(NC(=O)C=CC3CC3)C2)=O)CCCC2(CCCCC2)C1 C#Cc1cccc(C(=O)NC2(C)CCCN(C(=O)C(O)CSC)C2)c1F C12(CNC(C3CCN(C(C)=O)C34CC4)=O)COCCN1C(=O)OC2 Cc1cc(NC(=O)C(C)SC(C)C)c2[nH]c(C)c(C)c2c1 C(=O)(C(C)(C)S(C)(=O)=O)N1CC2C(CNC(CSc3nc(C)[nH]n3)=O)C2C1 C(c1ccco1)=CC(=O)NCCOCCOCCNC(C1CCSC1)=O CC(CO)N(C)NC(=O)C(C)CCOS(=O)(=O)N(C)C N1(C(C2(SC)CC2)=O)CCCN(CCCCNC(C2(C)CC(F)(F)C2)=O)CC1 c1(C(N2C(CNC(CC3N(C)CCC3)=O)CCC2)=O)cnc2ccccn2c1=O CON1CCC(CC(N2CC(N(C)C(c3nc(O)c(C)s3)=O)C(O)C2)=O)CC1 C(=O)(CC(C(F)F)n1cccn1)NC(C)CCCCNC(c1cc[n+]([O-])cc1)=O CCCC(C(=O)N1CC(CC(C)NC(c2cn(CC)nn2)=O)C1)NC(C)=O c1(C(N2CC(C(C)(C)O)(CNC(C(CC)O)=O)C2)=O)nnn(C)c1COC c1(CCC)ncoc1C(N1CC(O)(CCNC(c2ccn(C(C)C)c2)=O)C1)=O N1(C(C(=Cc2cccnc2)C)=O)CC(NC(=O)CNc2ncccn2)C(C)(C)C1 C(=O)(C1CCCc2cccnc21)NCCCC(C)NC(c1c(CC)oc(C)c1)=O CC1=NOC(CC(=O)N(CC(=O)NCCCc2ccncc2)CC2CC2)C1 N1(Cc2c(C)nc(CNC(=O)C(C)S(N)(=O)=O)o2)CCCNC(=O)C1CC(C)C N1(C(CCC#C)=O)CC2CCN(C(c3ccc(C(C)C)cc3Br)=O)C2C1 N1(C(CC(C)OC)=O)CCCC(CCNC(c2nnn(C)c2C(F)(F)F)=O)C1 Cc1cc(C)c(C(=O)N(C2(C(N3CC(CO)CC(C)C3)=O)CC2)C)cn1 N1(C(CN(C(=O)OC)C)=O)CCC(NC(c2ccc(-c3ccco3)[nH]2)=O)C(C)C1 C(=O)(CCCCC(C)(C)C)N1CC(NC(COC(CC)(C)C)=O)N(C)CC1 C1(N(C(=O)CC2CC3CCC2O3)C)CC2CCC(C1)N2C(=O)CC1CC=CCC1 C1(C(N2C(C(=O)OC)CCCC2)=O)CN(C(=O)C2=C(C)CCC2)CC(C)(C)C1 CCCC(C)(CCC)C(=O)N1CC2(C1)CN(C(=O)CS(=O)(=O)N(C)C)C2 C(=O)(C(C)C(F)(F)C(F)F)NC1C2(CN(C(c3n(CCC)nc(C)c3)=O)C2)CC1 Cc1ccc(C(C)CC(=O)NCCC(C)(C)CNC(c2csnc2C)=O)cc1 N1(C(Cc2cn(CC)nc2)=O)CC(NC(c2c(Cl)n[nH]c2C2CC2)=O)C(C)C1 C=CCCC(F)(F)C(=O)NCC(O)CCNC(=O)CCc1cc(OC)no1 CC1(C)CC(NC(c2cnc(CC(N)=O)s2)=O)CN1C(=O)CCNS(C)(=O)=O c1(C(N2CC(C)(CNC(CSC)=O)OCC2)=O)cnc2snc(C)c2c1 N1(C(CN(CCOC)C)=O)CCC(CCC(=O)NCCC(C)(C)OC(C)C)C1 C12(CCC(C)(C)C1)C(=O)N2C1CC1.Cc1cnccc1C(=O)NC1CCCC1 Cc1ccc(O)c(C(N2CC=CC(C(=O)NC3CN(C)CCC3O)C2)=O)c1 C1(CNC(COCCC)=O)(NC(c2sccc2C)=O)CC2CCC1CC2 N1(C(CCOCC)=O)CCN(C(=O)CSC(F)F)C2CCCCC12 C1(C)(C(N2CCC(CCC)CC2)=O)CN(C(C2CC(C3CC3)=NO2)=O)C(C)(C)C1 C(=O)(C(CC(C)(C)C)NC(c1cc(C)c(O)nn1)=O)NC(CN(CCC)CC)C C(=O)(CCN(OC)C(=O)C1CC2(CCN1C(=O)CCC1CCCO1)CC2)OC c1(OC(C)C(=O)N(CCCNC(=O)CC2CC2(C)C)CCO)cc(Cl)cc(Cl)c1 C1(CC=C)(NC(c2[nH]ccc2CNC(C2C(C(C)=O)C2(F)F)=O)=O)CCCC1 C1(NC(c2cc(C)c(C)s2)=O)CC2CC(NC(c3ccoc3C)=O)C1C2 Cc1nc2cccc(C(N3CC4C(NC(=O)C(O)C5CC5)C4C3)=O)n2n1 C(C(C)NC(c1cnc(C)n1C(F)F)=O)(C(C)C)NC(COCCCC)=O C1(NC(=O)C2=CCSC2)COC2(C1)CN(C(C13CCCC1C3(F)F)=O)C2 c1(NCCS(=O)(=O)N2CCCC2)cc(=NC2CCC2)[nH]c(Cl)n1 C(CCC(C)C(=O)NCc1cc(C)c(C(N2CCC(F)C2)=O)o1)OC N1(C(CCCCC=CC)=O)CCCN(C(=O)CC2C=CCC2)C(CO)C1 c1(CCC(=O)NCCN(C(=O)Cn2cc(C#N)cn2)C)c(F)cccc1F CCCCC(C(=O)NC(c1nccnc1C)C)NC(c1cc[n+]([O-])cc1)=O c1(C(N2C(C)CCC(NC(C3CC3C(N)=O)=O)C2)=O)c(Cl)ccc(F)c1N c1(C(=O)NC(COC)C(=O)NCCCC2CCOC2)ccccc1O C1(CC=C)(NC(=O)Cc2cncs2)CCCN(C(=O)CC2CCCCC2)C1 N1(C(=O)COCC2CC2)CC=CCC1C(=O)NCC1CC=CC1 C1(CN(C(CC(C)CF)=O)C)CN(C(=O)CCCCCc2cccs2)CC12CC2 c1(C(N2CCC(NC(c3cc(C)sn3)=O)CC2C)=O)ccc2c(c1)nnn2C C(=O)(CCC(CF)CF)NCCN(C(C1COCC1(C)C)=O)CC O=S(=O)(c1ccc(Br)cc1Nc1ncccc1F)N1CCC(C2CCOC2)C1 C1(NC(c2cccc(C(=O)NC)c2)=O)CCN(C(c2cnncc2O)=O)CC1C c1(C(N(c2cc(-c3ccc(Cl)s3)[nH]n2)C(C)C(=O)OC(C)(C)C)=O)ccc(Br)s1 c1(C(=O)NC2C(CNC(c3n(CC)ccc3)=O)CC2)cnc2[nH]cnc2c1 c1(C(N2CCCC(NC(CCC(=O)NCC)=O)C2)=O)cc(OC)nc(F)c1 C=CCC(C(=O)N1CCCC1C(=O)NCC1CCCC12CC2)NC(C)=O c1(OC)c(Br)cc(C(N2CC3CN(C(c4csc(C)n4)=O)C3C2)=O)cc1Br CC1C(NC(c2ccn(C)c2)=O)C(C)CCN1C(=O)CCCOc1cccnc1 c1(NC(C(C2CN(C(=O)C(F)CCC(C)C)C2)OC)=O)ccc(C)c(O)c1C c1(C(=O)OC)ccc(C)nc1NC(C1C=CCN1C(c1c[nH]c(=N)s1)=O)=O C12(CNC(c3cccc(F)c3F)=O)CCCCC1N(C(Br)Br)CC2 Cc1ncc(C#N)cc1NC(=O)C1=CC(O)C(NC(=O)CCC2CC2(C)C)C1 N1(C(c2c(C)noc2C(C)C)=O)CC2CCC(NC(=O)CC3CCOC3)CC2C1 C=CC(C)(C)CCCNC(C1C2CC2CN1C(c1ccc(F)cn1)=O)=O C1(NC(CC2C3CN(C(C#CC(C)(C)O)=O)CC32)=O)CCCCCCC1O N1(C(C)=O)CCOC2CN(C(c3csc(-c4nc[nH]n4)n3)=O)CC12 c1(NC2C(C)(CC)C2)ccc(S(=O)(=O)NCC2CN(c3ncccn3)C2)c(Br)c1 C1(C(=O)NCCC2CN(C(C(CC)N(CC)CC)=O)C2)C2CCCCC12 C(C(=O)OC)(C(C)C)(C(C)C)OC(c1ccc(C(=O)OC)c(C)c1)=O N1(c2ncc(C)c(C)n2)CCC2(CC1)CN(C(c1ccnc([N+](=O)[O-])c1)=O)C2 C1(C(C)NC(C=CSC)=O)CCN(C(=O)C(F)=CC2CC2)CC1 C1(C2C(=O)N2)CCC2CC1C2(C)C.C(C)(C(=O)OC)N1CC1.c1(C)ccco1.CO C1(C(C)=O)CCC(CNC(=O)NC(CC(F)(F)F)c2ccccc2)C1C Cc1ccc(C)c(C(N2CCCC2C2(C(N3CCOC(C)C3C)=O)CC2)=O)c1 C1(n2c(C(c3ccc(OCC)[nH]3)NCC)nnn2)CCCCCC1c1ccccc1 N1(CC)CCOC(C(=O)N(CCNC(C2(F)CC2C)=O)C(C)C)C1 c1(C(=O)Nc2cc(O)ncn2)ccc(S(=O)(=O)N2CCCCC2)cc1 Cc1oc(=NC(=O)c2cc(NCc3cccc4[nH]ncc34)cn2C)[nH]c1Br N1(C(C=CC=CCC)=O)CC2(CC(=O)N)CC(F)(C1)C2.C1(OCC)(OC)CCOC1 CC1(C)CCC(O)(C(N2CCCC(NC(=O)Cc3sccc3Br)C2)=O)CC1 C(CCCC(=O)N1CC(OCC(=O)NC2COCCC2C)C1)SC c1(C(N2CC(F)(CNC(C3(C)CCC(C)C3)=O)C2)=O)cc2n(n1)CCNS2(=O)=O N1(C(C(CCOCC)NC(CCCC)=O)=O)CC(O)(C2CCC2)C1 Cc1ccc(N2CCCC2)c(C(=O)N(CCNC(=O)C(O)C(F)F)C2CC2)c1 c1(C(N2CCCC2c2cccs2)C(=O)NC)ccccc1Br N1(C(C(=O)NC(C)C)=O)CC2CC(NC(c3cnc(C(C)C)nc3O)=O)CC1C2 C(C(C)CC(=O)NCCOCC(N1CC(O)(C(C)C)C1)=O)OC C1(NC(COC(C)(C)C)=O)CCCC1C(=O)Nc1ccnn1C1CC1 N=c1[nH]c(CCC(=O)NC2CC(CNC(c3sccc3Cl)=O)C2)cs1 N1(C(c2c(C#N)csc2)=O)CC(C2(NC(c3cscc3C(F)F)=O)CC2)C1 CCC(C)(COC)C(=O)NCCC(C)NC(c1ncccc1CSC)=O C(=O)(C1CCc2ccccc21)NCCCOCCNC(c1c(CC)n(C)nc1)=O N1(C(C2(COC(C)C)CCC2)=O)CCC(O)(C(C)CNC(=O)C(C(C)C)SC)C1 N1(C(C(CC)C2CCC2)=O)CC2(CC(C(=O)NCCCN3CCC3)CO2)C1 C1(C(C)(C)C)(NC(=O)NCCc2csc(C3CC3)n2)CCCC1 C#CCC(C(=O)NC(CC)C1CC1)NC(=O)CN=[N+]=[N-] C1(NC(=O)Nc2ccc(N3CCOCC3)nc2)CCc2nn[nH]c2C1 c1(CC(=O)NC(CCNC(C(CC)(C)F)=O)C)ccc(Cl)cc1F c1(SCCOC(c2ccc(-c3ccncc3)cc2)=O)ccc(Br)cc1 O(C1CCCc2ccccc21)CC(=O)NC1CCC(NC(CC=CC)=O)C1 N#Cc1cc(C(=O)OC2CCC(C#N)C2)cnc1-c1ccccc1 c1(C2C(C(=O)NC(C3CCN(C(c4cnco4)=O)C3)C)C2)cccnc1 c1(C(N(CC(CC)NC(c2cnn(C)c2C(F)F)=O)C)=O)ccn2nnnc2c1 CCC(C)CCC(=O)NCC(C)CNC(=O)COc1ccccc1C N1(C(CC=C)=O)CCN(C(=O)C(C)(C)C(=O)OCC)CC(C)(C)C1 N1(C(C(COC)O)=O)CC(C)(C)OCC1CNC(c1c[nH]c(=N)s1)=O N1(C(CCCC(C)(F)F)=O)CCCC2CN(C(C3(N(C)C)CCC3)=O)CCCC12 C#CCC(C)C(=O)N(c1ccccc1OCC(=O)OCC)C(C)Cc1ccco1 C(=O)(C(F)(F)C(O)C(C)C)NC(CCNC(C1(CCOCC)CCC1)=O)(C)C C1(C(CNC(c2cc(OC)ns2)=O)(C)O)CCN(C(C2CCC(=O)O2)=O)CC1 c1(C(N2CC(CC(C)NC(CC3C(CC)C3)=O)C2)=O)cc(O)cc(C#N)c1 C(=O)(C(CC(=C)C)OC)N1CC(CC=C)(C(=O)NC(c2cnn[nH]2)C)C1 n1(CCCC)ncc(C(=O)NC2CC(O)(CNC(C3CC=CCC3)=O)C2)c1C C1(CC)CN(C(c2conc2CNC(=O)C(C)(C)C#N)=O)C(C)CO1 C1(NC(COCc2cccc(C)c2)=O)CN(C(=O)CC2CC2(C)C)CC2(CC2)C1 c1(C(=O)NCCOCCCF)ncccc1Cl C(=O)(C(F)C(C)(C)O)NC(CC=CC)C(=O)N1CCCCC1CC(N)=O C(=O)(CCCCCS(C)(=O)=O)NC(C)CC1CN(C(=O)Cn2nnc(=O)[nH]2)C1 c1(COC)nc(CC(=O)N(C)CC2CCN(C(c3cc(C4CC4)no3)=O)C2)cs1 C(CC(C(=O)N1CCOC(C2CC2)C1)NC(=O)CC1CC(C2CC2)C1)OC c1(C(C(=O)NC(C)CC(C)NC(C2CC2C)=O)OC)c(Cl)cccc1Cl N1(C(CCC(C)OCC)=O)CC=C(C(=O)NC2(C(C)C)CCC2)CC1 C12(C(=O)NCC3CC(NC(C4(C)CC(OC)(OC)C4)=O)C3)CC(C1)C(C)(C)O2 c1(CC(=O)NC2C3CN(C(C4(C)CCN(C)C4)=O)C2C3)cccc(F)c1F CCC(C)(CNC(C1CCC(C)(C)OC1)=O)C(=O)NCCN1CCCC(O)C1 c1(CCC(N2CC(COC)(NC(c3cc(Cl)n(C)n3)=O)C2)=O)cnc(C)nc1O C1(OC)C(C)(C)CN(C(=O)C(c2ccc(F)cc2)C)C1(C)C CC1CCC(C(C)(C)C)N1Cc1ccncc1-c1cc[nH]c(=N)c1 C1(NC(Cn2ccc(C)n2)=O)CN(C(=O)Cn2nnc(=N)[nH]2)CCC1F CCCC(C#N)C(=O)NCC(F)CNC(c1nnc(O)cc1O)=O CCCCC(C)(F)C(=O)NCc1ccc(C(=O)NCC2CC2(Cl)Cl)cc1 C(=O)(C1=Cc2ccccc2C1)NC1CCN(C(C=C2CCC(C)CC2)=O)C(C)C1 N1(C(CC(COC)(C)O)=O)CCN(C(c2cnc(CC3CC3)s2)=O)CC(C)(C)C1 C1(NC(=O)Cc2ccc(O)cn2)CN(C(=O)C2=CCC2)CC2(CCC2)C1 N1(C(C2N(C(CCCC#CC)=O)C3C(C2)C3)=O)CCCC2(CCCO2)C1 C1(C(=O)NC(c2cn(CC)nc2)C)CN(C(=O)CC2COCCO2)C(C)(C)C1 c1(C(=O)NCC2CCC(NC(C3N(C)CCC3)=O)CC2)cc2ccncc2[nH]1 Cc1c(C(=O)NC2(C)CCCN(C(=O)CC3COCC3(C)C)C2)nn(C)c1N c1(C(=O)NCC2C=CC(NC(CCOC(C)C)=O)C2)nccn2ccnc12 Cc1ccc(=N)[nH]c1CC1CCCC1.N1(CCC(=O)NC(CN)C)CCCCC1C C1(C(=O)NCC2CCN(C(Cc3c(C(C)C)con3)=O)C2)CSCC(=O)N1 C=CCCCC(C(=O)N1CCCC(N(C)C)C1)NC(c1ncc(F)cc1F)=O c1(COC)ccc(C(=O)NC(C2N(C(C3(N(C)C)CC3)=O)CCC2)C)o1 N1(C(Cc2cccc(C)c2)=O)CCC2C1CCN2C(=O)Nc1cc(Cl)ccc1C C1(NC(Cc2cc(C)no2)=O)CCN(C(=O)Cn2nccc2C)C12CCCC2 C12(C(N3CC(C(C)NC(=O)Cn4ccc(CO)n4)OCC3)=O)CCC(CC1)CC2 C=C1CCC(C(=O)NCCC(O)CNC(c2cccc(C(F)F)c2)=O)CC1 c1(C(N2CCN(C(CC)C(N)=O)CC2)=O)cc2c(C)cccc2o1 C(=O)(CCC(C)(C)C#N)NCC(CC)CC.C12(CSC1)C(=O)N2CC CCC(C)CC(C(=O)NCCCF)NC(=O)C(C1CC1)CCOC c1(C(C(=O)NCC2CC2)N(C2(C)CCCC2)CC(=O)OCC)ccnc(OCC)c1 C1(CN2CC(C(=O)OCC)C2)CCCC1(C)C.N12CC(C)(C1)C2=O c1(OC)cc(O)c(C(N2CCC(O)(CN(C)C(C)=O)C2)=O)cc1OC c1(C(C(=O)NC2CC(NC(C3CCC(C)C3)=O)C2)(C)C)ccc(Cl)cc1 C1(CNC(c2ccc(CC)c(CC)c2)=O)CCN(C(C2CCCC2)=O)C(C)C1 C(=O)(CS(=O)(=O)C1CCCC1)N1CC2N(C(C(CC(C)(C)C)(C)C)=O)C(CC2)C1 c1(CNC2CCC(C(=O)NCCC3C(C)CCC3)C2)ccc(C#N)s1 Cc1nn(CC(N2CC(CNC(c3cnns3)=O)CC2C)=O)cc1Br c1(C(=O)OC(C(=O)Nc2c(O)ncc(C)c2)C)cc(O)c2nc(C)n(C)c2c1 C=Cn1nccc1C(=O)NCC1(CCN(C(=O)C(O)C2CC2)CC)CC1 C1(CC(=O)N(CC(F)F)CC2CC2)CCCN(C(=O)CCN2CCCCC2)CC1 N1(C(CC2(N(C)C(C3CC3C3CC3)=O)CC2)=O)CC(CO)C(CO)C1 N1(C(CC=CC=C)=O)CCC(C(C)C(=O)NCCS(C)(=O)=O)CC1 C#Cc1cccc(C(=O)NC2CN(C(c3cnnn3C3CC3)=O)CC2O)c1F c1(CC(=O)NCC(CC)(C)NC(c2ccc(C(F)F)cc2)=O)ccc(Cl)nc1 c1(CC(=O)NCCCC(C)NC(CCC)=O)ccc(F)c(Cl)c1 CC(C)CCC(F)C(=O)N1CC(CNC(=O)C(=Cc2cscn2)F)OC(C)(C)C1 c1(CCOC(=O)NCCOCC=C)cnn(C)c1 CC1OCCC1CNC(=O)Cn1cc(CNC(C2CC23CC3)=O)nn1 C(=O)(C(C)C(C)NC(C1CCC1OC)=O)N(CC)Cc1ncc[nH]1 C1(C(=O)NC(c2c(C)cccn2)c2ccccc2)(CN)CCCCCC1 C1(NC(CC(C)C(F)F)=O)CC12CCN(C(=O)C(C)(C)CC#N)CC2 C(CN=C1NCC2(CCOCC2)NC(=O)CN1)OC.C1(CSC)CC=CCC1 CCC1CN(C(=O)C(C)NS(C)(=O)=O)C(=O)N(C)CC(=O)N1.C(C)(=O)OC C=CC1OCCC1C(=O)NC(C)(CNC(=O)CCc1ccc(O)nn1)CO CC1C(C(=O)NCC2(N(C)C)CC2)C(O)C(=O)N1C.C12CC(C1)C(=O)N2 N1(C(CCC(C)(C)F)=O)CCC2(COC(CNC(=O)CCCCCF)C2)C1 N1(C(CC(C(C)C)C)=O)CC(NC(c2ccc(CO)cc2F)=O)CC(C)(C)C1 N1(C(C(C(C)OC)OC)=O)CCN(C(=O)CS(=O)(=O)CC2CCCO2)CC1CO c1(C2C(C(=O)NCc3c(C(=O)NCC(C)O)cco3)C2)cccnc1 C1(CC=C)(NC(c2cncc(N)n2)=O)CCCN(C(c2ncc(C(F)F)s2)=O)C1 N1(CC(N2CCOCC(NC(c3nc(CC)oc3)=O)C2)=O)CCc2ccccc21 N1(C(C2(C)CC(F)(F)C2)=O)CCC(NC(=O)CCC2CCCC2)CC1C1CC1 Cc1cc(C(=O)NC23CC(C2)N(C(=O)CS(C)(=O)=O)C3)cn(C)c1=O Cc1ccc(C(N2CC3CC3C2C(=O)NCCn2ccnc2)=O)c(O)n1 c1(C(=O)NCC2(F)CC(NC(CCOCCOC)=O)C2)ccc(Cl)cc1C C(CC(C)CC)(C(=O)NCC(C)(C)C1(O)CCC1)NC(C(CC#C)C1CC1)=O C1(CNC(C(C2CCC2)OCC)=O)CCCCN1C(=O)CC(C)N(C)C C1(C(N2CCN(CCF)CC2)=O)CC2(CC2)CN1C(c1cc(Cl)ncc1Br)=O C1(NC(C2(CCCC)CCCC2)=O)CC(C)N(C(=O)CN(CC(=O)NCC)C)C1 c1(N2CC(CCNC(C3(CC)CC3)=O)S(=O)(=O)CC2)[nH]c(=O)n(C)c(=O)c1C#N CC1(C(N2C3CSCC2C3)=O)C#CCCCCCC1.c12ccc(cc1)c(=O)[nH]2 c1(CC)noc(C)c1C(N1CCN(C2CN(C(=O)Cc3n[nH]cc3Br)C2)CC1)=O N1(C(c2cccc(OCC)c2)=O)CC2CC(NC(C3(C(=O)NC)CC3)=O)CC2C1 c1(C(N2CC(CC(C)NC(c3c(CC)scc3)=O)C2)=O)ccc(Cl)c(F)c1N c1(C(=O)NC(C2CCCN2C(C2COCCO2)=O)C)cc(S(C)(=O)=O)co1 CN1CCC(C(=O)N(CCCNC(=O)C(C)(C)C2CCC2)C2CC2)C1=O N1(C(C(CNC(=O)CCOCCN(C)C)NC(N)=O)=O)CCCC(C)C1.CC(C)O C(C(=O)N=c1c(Br)c[nH]cc1Br)C1N(Cc2c(C#N)cccc2)CCOC1 C1(O)(CNC(C(CCC)c2ccccc2)=O)CCCN(C(=O)Cc2cc[nH]c2)C1 C1(C(=O)NCC(C(=O)NC)C)CCN(C(C2CN(C)CCO2)=O)CCO1 c1(CC)nc(NC2CCCn3ccnc32)nc2cccc(F)c12.C1CC1C1CC1N N(C(=NCCCF)NCC1(C)COCCO1)CC(C)CN1CCOCC1 N1(C(CC=CC=C)=O)Cc2ccccc2C(NC(=O)CN2CCC(F)(F)C2)C1 C(=O)(C1CCc2c[nH]nc21)NC1C(CC)CN(C(=O)CN(C)CCSC)CC1 N1(C(C2(C(C)NC(C3CCC(C4CC4)C3)=O)CC2)=O)CC2(C)COCC2(C)C1 C12CCCCCCC1NC2=O.c1(OC(COC)C)cccc(C(=O)OC)c1 c1(OC)ccc(C(CNC(=O)C(C)(C)c2cnsc2)NC(=O)C=CC2CC2)cc1 c1(CC)nccnc1NC(c1cc(NC(c2cc(C)nn2C)=O)cn1C)=O CCC1=C(C(=O)N(C2CC3CCC(C2)N3C(=O)CC2CCN(C)C2)C)SCCO1 C1(C(=O)NCc2cccc(NC(C3(C=C)CCCC3)=O)c2)CCC2C1C2(F)F N1(C(C2OCCN(C)C2)=O)CC(NC(=O)C=Cc2cn(C)cn2)CC(O)C1 C1(NC(c2c(OC)nccc2)=O)CC2CCC1CN(C(=O)Cn1[nH]cnc1=N)C2 CC1OC2CCC1(C(N1CCC(NC(C3CCC(C)(C)O3)=O)CC1)=O)C2 CC(=O)CCCC(=O)NCC(C)(C)CC(=O)NCC12CCCCC1C2 c1(NC(CSCC(=O)N(C)C)=O)cccc(C(=O)NC2CNC(=O)C2)c1 CCC(CC)C(F)C(=O)N1CCCC(N(C(c2[nH]cnc2C)=O)CC2CC2)C1 N1(C(c2cnc(C)n2C(F)F)=O)CCCC(n2cc(N(C)C3CC3)nn2)CC1 c1(C(=O)NC(C)(CNC(=O)CCCC(F)F)C2CC2)cc(O)nc2ccccc12 Cn1ncc2c(NCCC=CBr)[nH]c(=NCC3CCOCC34CCCC4)nc12 N1(C(=O)C(=O)NC(C)CC(=O)N(C)C)C(CO)CC1C.CCN c1(C(C)C(=O)NC2CC(NC(=O)CCCNC(=O)C3CC3)C2)ccc(F)cc1 C=CC(CCC)CC(=O)N(C)CC1CCN(C(c2oc(CC)cc2C)=O)C1 C1(CNC(c2cncc(OC)c2)=O)CC12CCN(C(=O)C=CBr)CC2 C1(C)(NC(CCOCCCNC(C(C)OC(C)=O)=O)=O)CC2CCC1C2 Cc1cccc(OCC(=O)NCC2CC3(CC3)CN2C(C2CCCSS2)=O)c1C C1(C(=O)NC(CCCNC(Cc2c(C)noc2)=O)C)CC12CC(OC(C)(C)C)C2 Cc1nsc(N)c1C(=O)NC1CC(NC(c2cnc(C(F)F)s2)=O)CC1O C(=O)(C1CCc2nccn21)NC1C(CNC(c2ccc(C)c(C#N)c2)=O)C1 c1(OC)cc(O)cc(O)c1.c12ccccc1-c1cnc(nc1)Cn1ccnc1-2.CCS C(=O)(CC(CN(C)C)CC)NC1CN(C(c2cccc(CC)n2)=O)CC1C n1(CC)ccnc1C(c1nnnn1C(C)(C)C)NC(C)C.C1CC(=O)N1 c1(C(N2CCC(CC)(NC(c3ccc(F)s3)=O)CC2)=O)cc2cccnc2cn1 c1(C(C)(F)F)cc(C(=O)NC2CC(C)(CNC(=O)CC3CCN(C)C3)C2)ccn1 C1(NC(Cc2c(C)noc2C)=O)CS(=O)(=O)CC1NC(c1cn(C)nc1Cl)=O N1(C(CC#C)=O)CC2CN(C(=O)C(C)NS(=O)(=O)CCCC)CC2C1 C1(CNC(c2cnc(C)nc2C2CC2)=O)CCC(C)(C)CN1C(C1CC1(Cl)Cl)=O C1(C(=O)OC)(C(=O)NCC(C)NC(C2CN(C)CC2C(F)(F)F)=O)CCCCC1 CC(C)CCC(O)C(=O)N1CCOCC1CCNC(=O)Cn1ccnc1C(C)C CC1(C(=O)NCC2CC2C(N2CC(n3cnnc3)C2)=O)CC2CC2C1 c1(C(C(=O)NC(CCNC(C(C)(C2(C)CC2)OC)=O)C)C)c(C)noc1C n1(CC=C)c(N2CCCC(C)C2)nnc1CCn1ccnc1C.OCC C(CC(C)C)(C(=O)NCC(O)CC(=O)NC)NC(C(C)OCCC)=O CC(CC(F)(F)F)C(=O)NC1CC(C)(NC(c2cnn(C)c2)=O)C1 c1(C(=O)NCC2N(C(CC3(CC)CCC3)=O)CCC2C)cc(C)cc(Cl)c1O C1(NC(=O)CC2CCS(=O)(=O)C2)CN(C(C23CSC(C2)C3)=O)CC1C1CC1 c1(C(N2CCN(C(c3cncnc3)=O)CC2)=O)ccc2c(c1)CCO2 c1(C(C(=O)NCC(CN(C(C2(c3c(C)ccs3)CC2)=O)C)C)C)cccc(F)c1 c1(C(=O)NCC2C(C)(C)CN(C(C3CC34CC4)=O)C2)cc2ccc(Br)cn2c1 c1(C(c2nnnn2C2CC2)NCCSCC)csc(C(F)F)c1 CC(C)(O)C(F)(F)CNC(=O)C(Cc1ccco1)NC(c1cc[n+]([O-])cc1)=O C1(CC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)COCC(C)C c1(C(=O)NCCCCN(C(C(CC2CCC2)OC)=O)C)ccc2nccn2c1 C1(NC(C2(NC(C)C)CC2)=O)CC2CCCC(C1)N2C(C1CC(C)C1)=O c1(N2C(C)CC(NC(CCC(=O)NCC)=O)C2)nc(C(F)(F)F)ccc1C#N c1(C(N2CCC(NC(C(CCC)C)=O)C(F)C2)=O)ccc(F)c(C#N)c1 c1(C(C)C)c(N2CCC(CF)(NC(=O)C(C)Cc3cnn(C)c3)C2)ncnc1Cl C(CCCC(=O)N(C1CCN(C(c2cncnc2C(C)(C)C)=O)C1)C)SC c1(C(=O)NC(Cn2cc(C(=C)C)nn2)C)cc2cc(Cl)ccc2n1C N1(C(C(CC)OCC)=O)CC=C(CNC(c2c(Br)nnn2C)=O)CC1 N1(Cc2ncc(C)nc2)CCN(c2ncc(C(F)(F)F)cn2)CC1C NC(=NCCCF)NCCC(C)(F)F.CCC(C)(C)O Cc1c(F)ccc(N)c1C(=O)NC1CN(C(=O)CC2CCCCC2O)CC1(C)C C1(CC(=O)N(C2CCN(CC)C2)CC)CCCC12CC2.C1(=O)CC2(CC2)N1 c1(C(=O)NCC2(F)CC(CNC(C3CC4CC4C3)=O)C2)ccc2snnc2c1 c1(OC)cncc(C(N2CCC(NC(=O)C3=CC(C)(C)C3)C2C(C)C)=O)c1C C1(N(C(Cc2c(C)nc[nH]2)=O)C)CCC2CN(C(c3ccn(C)c3C)=O)CC12 C1(C(N(C)C2CC2)=O)CC12CCN(C(=O)C(C)(C)C1CCC1)CC2 C(=O)(CCS(C)=O)NCC(COC)NC(c1cncc(OC(C)C)c1)=O C(=O)(C(C)(F)C(F)(F)F)NC1C(C)CN(C(C2CC2c2ccco2)=O)C1 N1(CCC(N2C(C3(NC(C4CCC45CCC5)=O)CC3)CCC2)=O)CCCCC1=O C(C(O)CNC(=O)CC1CCCC1)N(C(=O)CCNC(c1cccs1)=O)C CCC(C)C(C(=O)NCC(=O)Nc1ccc(CC(C)C)nc1)N(C)C C(=O)(CS(C)(=O)=O)N(C(CC)C(=O)NCCc1cocn1)C c1(CN2CCCC(C(C)NC(C(CC)CC)=O)C2)ccc(S(=O)(=O)N(C)C)s1 C(=O)(C(O)CCC(C)C)N1C(C(=O)NCc2ccc(CC)o2)CN(C)CC1 C(=O)(CC(C)(C)C)N(C(C)C)CCNC1CCCCO1.C1(c2ccon2)C(=O)N1 C1(F)(CNC(C=C(C)Cl)=O)CCCN(C(=O)CN2CC3CCC2C3)C1 c1(CC(C(N2CCC(COC)CC2)=O)N)cc(C)cc(F)c1 C(C)(CC(C)CC)N(C(C1(NC(COCCCC)=O)CCCC1)=O)C N1(C(c2cc(CC)sn2)=O)CCN(C(c2ccc(F)c(C)c2)=O)CC1CC c1(-c2ccn(C)n2)cn2c(n1)CCC(C(=O)Nc1cc(CO)ccc1C)C2 C1(NC(C2N(C(C(c3cncnc3)C)=O)CCC2)=O)CN(C)CC1C C1(N(C(c2c(C)con2)=O)C)CCCN(C(=O)C=Cc2cn[nH]c2)C1 c1(C(=O)NCCC2OCCN(C(Cn3nnc(=N)[nH]3)=O)C2)nnn2c1CCCC2 c1(OC)cc(Cl)ccc1C(=O)N(C(C)CCNC(=O)CCCOC(C)(C)C)C c1(CN2C(C(N(CCCCC=C)C)=O)CC(C)C2)cc(Br)c(NC)cc1C c1(C(N(CCCNC(C(n2cnc(C#N)n2)C)=O)C)=O)cc(=O)cc(Cl)[nH]1 N1(C(C2(C(C)(C)O)CC2)=O)CC2=C(C1)CN(C(=O)Cc1ccc(Cl)c(F)c1)C2 C(=O)(C(O)C(C)(C)C)NCC(CC(C)C)NC(C1C(C)(C)C1(F)F)=O C(=O)(CC(C)CC(C)C)N1CC(SCC)C(NC(C2(C)CC3C=CC2C3)=O)CC1 CC1CCC(OCC(N2CC(C(N)=O)(CNC(C3COC(C)(C)C3)=O)C2)=O)CC1 N1(C(CCCOCC)=O)CCC(CCC(C)(C)NC(c2ncncc2Cl)=O)CC1 Cc1c[nH]c(CSc2cccc(Cl)c2)c1C c1(C(=O)OCCC2CC2)c(F)ccc(S(=O)(=O)CC2CC2)c1F C1(C(=O)NCC2(NC(=O)CCn3cc(C)cn3)CCCCC2)(OC)CS(=O)(=O)C1 c1(C(=O)NC(CC)CN(C(=O)C(F)OC(F)(F)F)C)c(C)csc1Cl c1(Cn2cc(CNC(=O)CNC(c3cccc(=O)o3)=O)nn2)ccc(F)cc1 CON(CCC(=O)NCC1CCOCC1C)C(=O)CC(C)(F)F CCCCC(O)C(=O)N1CC2CC1C2C(=O)Nc1cncc(Cl)c1 N1(C(c2ccc(C)c(O)c2)=O)CC(NC(C23CCCC(C2)OC3)=O)CC(C)(C)C1 N1(C(c2cc(C)c(F)cc2)=O)CCC2(NC(c3cscn3)=O)CCCC12 C1(C(=O)NCC(C2CCCC2)C)CN(C(=O)Cn2c(O)nnc2O)CCN1C C1(C(N2CC(C)(C(=O)NCC(C(C)C)C)C2)=O)CCOC(=O)CC1 C1(CN(C(C(N2CCOC2=O)C)=O)C)CN(C(=O)C(O)(C2CC2)C2CC2)CCO1 c1(CNC(C2COCCN2C(C2(CO)CC2)=O)=O)csc2ccccc12 c1(C(=O)NCC(CC(F)(F)F)NC(COCC)=O)nn(C)c2ccccc2c1=O C=CC1(CC(=O)NC2CN(C(c3cnnnc3C)=O)CC2F)CCOCC1 C1(O)(CC#N)CCCN(N2CCC(C(N3CCOCC3)=O)CC2)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)COC2(C)CCCC2)ccn2c1CSCC2 N1(CC(C)NC(N)=O)CCN(C(=O)Cc2cccc(OC(=O)C(C)(C)F)c2)CC1 CC1OC2CCC1(NC(C1CC(NC(c3cccs3)=O)C1)=O)C2 CCCCC(CCCC)NC(=O)CC(CC1CC1)NC(=O)C=CC(C)CC CCC(C)(C(=O)N1CC(O)(CNC(c2cc(O)cs2)=O)C1)C(F)F CC1CCC=C1C(=O)N1CCCC(n2cc(C(NS(N)(=O)=O)(C)C)nn2)C1 c12csc3nc(nc(O)c13)N(C)CC2.C1(CC(=O)NC(COC)C)CCC(=O)N1 C(C)(C)(CC(C)NC(=O)NC(c1cccc(C(F)F)n1)C)OC Cc1cc(N)c(F)c(C(=O)NCC(C)(C)NC(c2nc(O)c(C)s2)=O)c1F N1(C(C2(CC)CCOC2)=O)CC(CO)C2(C1)CN(C(c1csc(C(F)F)n1)=O)C2 c1(C(=O)NCC2C(C)(C)C2C(=O)NC2CC23CCC3)ncnc(O)c1F C1(C2CCN(C(C3(Cl)CC3C(C)=O)=O)CC2)(C(=O)NC(C#C)(C)C)CCOCC1 c1(C(=O)NC2CCCCN(C(CS(C)(=O)=O)=O)C2)ccc2c(c1)CCC2=O CCC(C)C(O)C(C)C(=O)NCC1(F)CCN(C(c2cc[nH]c2C)=O)C1 C1(CNC(CC)=O)(COC)CCN(C(c2ccc(CO)cc2OC)=O)CC1 n1(CC(N2CC3C(CNC(c4coc(CO)c4)=O)C3C2)=O)ccc(Br)cc1=O N1(C(N(CC(C)N(C)C)CC)=O)CC(C2CC2)C(F)(c2ccccc2)C1 Cc1ccc2cc(C(=O)N(C(CNC(=O)CN=S(C)(C)=O)C3CC3)C)cn2c1 C1(NC(C2(OCC)CCSCC2)=O)CC2CCC1N(C(c1ccnn1C)=O)C2 c1(C(=O)NC2(C)CCN(C(C3CCCC3(F)F)=O)C2)cc(F)c(F)cc1Br C#CCCCCCC(=O)C(CCCCN(C)C)C(=O)NCCCCCCCNC N12C(CC3CCCCC13)C(=O)NOCC(=O)NCCC(O)C2=O.C(C)(=O)OC c1(CNC(C(C)(C)NC(C2C(C)C2C)=O)=O)cncc(F)c1 Cc1cc(Cl)nc(Cl)c1NC(C1CC1C(=O)Nc1ccc2nncn2c1)=O C1(OC)CN(C(c2ncc(C)o2)C(=O)NCC(F)F)C(C)(CO)C1 N1(C(c2c(C)nc[nH]2)=O)CCCC(N(C)C)CC1.c1(CC(=O)NC)ccccc1F n1(CC(N2CC(CNC(C(CC)C)=O)(OC)C2)=O)cnc2sccc2c1=O c1(C(c2cccc(F)c2)NC2CC(NC(=O)OC)C2)cc(Cl)c(CO)c(Cl)c1 CON(C)CCCNC(C1(CNC(c2nnsc2C)=O)CC2(CC2)C1)=O C1(C(=O)NC)CCCCN1C(C12CC(NC(=O)CCc3ccccc3)(C1)C2)=O C1(CNC(c2ccn(CC)n2)=O)COCCN(C(=O)CC2CCC(=O)O2)C1 c1(OC)ccc(CC(=O)NC2(C)CCN(C(C3CC3(C)C)=O)C2)c(OC)c1 CCCC(C(=O)NC(c1cn(C)nn1)C)NC(=O)CNC=O c1(C(=O)NCC2(O)CN(C(c3cc(C(C)=O)oc3C)=O)C2)cnc2occc2c1 c1(OC)ccc(CNC(=O)C(N2CCC(CO)CC2)c2csc(C)n2)c(OC)c1 Cc1ccc(-c2cccc3c(NC(=O)C4CC4)c[nH]c23)c2n[nH]cc12 c1(CC)nccn1C(C)CC(=O)N1CCC(NC(=O)COc2ccon2)C1 c1(OC)nccc2cc(NC(=O)NCC3(C4CCOCC4)CC3(F)F)ccc12 N1(C(CC(C=C)C)=O)C2CCC1C1CC1(NC(=O)CNC(=O)C(C)(C)C)C2 n1(CC)nnc(C(=O)NC(C2CCN(C(=O)CC3CC4CC4C3)C2)(C)C)c1C C1(C(=O)NCC2CC2)CN(C(=O)CNC(C2(C)CC2)=O)CCC1F.C(CCCl)S C1(C(=O)NCC2C(C)OCC2)CN(C)CCN1C(C1CN2CCC1CC2)=O N1(C(c2c(C)noc2)=O)CCCC(O)(CNC(C2CC2C2CC2)=O)CC1 C(CCCCCS(=O)(=O)CCO)NC(c1ncc(C)s1)C1CC1 C(=O)(C1=COCCC1)N1CC(C)(NC(c2ccn(C3CCCCC3)n2)C2CC2)C1 c1(OC)ccc(C(C)C(=O)NCCN(C)C(C2CC=CCC2C(F)(F)F)=O)cc1 N1(C(C2(CC)CCOC2)=O)CCCN(C(=O)CCn2cc(Cl)cn2)C(C)C1 c1(C(N2CCN(C)CC2)C(=O)N(CCC2(C)CC2)C2CC2)cn(C)nc1Br CCC(C(=O)NCCCC(C)NC(c1n[nH]c2ccccc12)=O)C(F)(F)F Cc1nc(CC(=O)NC2CCC(CNC(C3CCCC34CC4)=O)CC2)cn1C C(C(C)(C(=O)NCCc1cnccn1)NC(=O)C(C1CCOCC1)F)SC c1(OCCOC)cccc(NC(=O)CN2CCC(NC(C3CS(=O)(=O)C3)=O)C2)c1 C(=O)(CCCN1CCCCC1)N(C(C)CNC(c1coc(COC)n1)=O)CC C12(CNC(CC#N)=O)CCC(NC(c3cc(CCO)on3)=O)(CC1)CO2 N#Cc1ccc(N)c(C(=O)NC2CC3CCC(C2)N3C(c2cccnc2S)=O)c1 c1(C(N2CCC(N(CC#C)C(c3nccs3)=O)CC2)=O)ccc2c(c1)CCN2 c1(C(=O)NC(C)CCCNC(=O)CC(c2ccccc2F)C)n[nH]c2c1COC2 CN1C(=O)c2ccccc2C1CC(=O)NC1C2CC1CN(C(=O)CS(C)(=O)=O)C2 C(=O)(C1=CC2CCCCCCC12)NCC(C1CCOC1)NC(=O)CN1CCC1 N1(C(CCC(C)C)=O)CCCC(NC(C2CCN(c3ncccn3)C2)=O)CC1 C1(C(=O)NC2CCN(C(c3onc(C)c3C)=O)CC2O)CC(C)(C)OC(C)(C)C1 CC(C)C1=NOC(C(N2CCN(C(c3ncnc(O)c3Cl)=O)C(C3CC3)C2)=O)C1 c1(C(N(C(CN(C(C(CCOC)C)=O)C)C)C)=O)cc(Cl)c(F)cc1F C(N=c1ccc(-c2cccc(C#N)c2)n[nH]1)C1C(C)CCNC1=O N1(C(c2cccc(=O)o2)=O)CCOCC2(COCCN2C(=O)CCCCCF)C1 C1(CC=C)(C(=O)NCc2cc(C)nn2C)CCCN1C(=O)Cc1cn(CC)nn1 C1(C(=O)NOCC2CCOC2)N(C(c2cc3n(n2)CCC3)=O)CC12CCCC2 c1(CC(CNC(=O)CCc2cnoc2)NC(C2(CC=C)CCC2)=O)ccccc1 C1C(C)(C)C(=O)O1.c1(COCCOC)cccc(NC(=O)OC(C)(C)C)c1 C1(CN(C(Cn2ncc(C)c2)=O)C)CCCCN1C(=O)C(C1CCC(=O)N1)C Cc1nn(C)c(C)c1C(C)C(=O)N(C(C)CNC(c1nccnc1N)=O)C c1(OC)ccc(Cl)c(C(=O)NC2COCCN(C(=O)CS(=O)(=O)N(C)C)C2)c1 C1(NC(CSCCC)=O)CN(C(c2scnc2C(F)F)=O)CC1OC C1(NC(C(C)C2CCC2)=O)CCC12CCN(C(=O)CCc1ccc(O)nn1)CC2 N#Cc1ccccc1C(N1CCN(C(C2CCCS2(=O)=O)=O)C2CC12)=O CON1CCC(C(=O)NCCOC(C)(C)CNC(c2cnc(C)c(N)c2)=O)CC1 c1(C(=O)NCC2CC(NC(=O)Cn3ncnn3)CC2O)coc2c1COC2 N1(C(CSCC=C)=O)CCCC(N(C)C(C2CN(C)CCO2)=O)C1 CC1(C)C=C(C(=O)NCC2COCC2NC(c2cc(-c3cccnc3)no2)=O)C1 C(=O)(C(C)(O)C(F)(F)F)NCCC(C)N(C(c1c(CC)nns1)=O)C CC1CCCN(C(=O)C=CC2CC2)C1CNC(c1ccnc(OC(F)F)c1)=O C#CCC(CC(=O)Nc1cncc(C2CC2)c1)NC(c1cnn[nH]1)=O C12(C(N3CCC(N(C(=O)CN(C)C4CC4)CC)C3)=O)CCC(F)(CO1)C2 Cc1ccccc1C=CC(N1CCC(NC(=O)C2=CCOC2)C1)=O CC(C)(C)C#CCCNC(C1CC1CNC(=O)COc1ccccc1)=O C(C1CCCCC1)=CC(=O)NC1CCN(C(=O)Cc2cc[nH]n2)C1C1CC1 C1(C(=O)NC2C=CCN(C(c3nc(C(=O)OC)oc3)=O)C2)CCC(C)(C)OC1 c1(C(C)C)cc(NS(=O)(=O)CC(N)=O)c(O)c(C(C)C)c1.N12CC(C(C#N)C1)C2 C(=O)(CC(F)(F)CC(=O)N1CC(NC(C2CCOC(C)(C)C2)=O)C(C)(C)C1)OC c1(C(=O)NC(CNC(COCc2cc(C)no2)=O)(C)C)cc(N)ccc1Cl N1(C(=O)COC(F)(F)F)CCC2OCCN(C(c3cc(CO)cc(F)c3)=O)C2C1 C1(NC(C2CCN(CC)C2)=O)CN(C(=O)C(Cl)(Cl)Cl)CC12CC2 N1(C(c2n(CCC)ncc2)=O)CCC(NC(c2nccc(SC)n2)=O)C(CC)C1 Cc1cccc(C2CC2C(=O)NCC2(F)CN(C(c3c(Br)n[nH]c3C)=O)C2)c1 Cc1cccc(NC2CCC2)c1C.c1(CNCCC#N)sc(Br)nc1C C1(NC(C2N=C(C)SC2)=O)CC2(CCCN(C(c3ccc(C)[nH]3)=O)C2)C1 Cc1ncc(C(C(=O)NC(C)(C)C)N(C2CC2)Cc2nncn2C)[nH]1 C1(C(N(CCCNC(=O)CC2(N(C)C)CC2)C)=O)CCC1F C(=O)(C1=NOC(CO)C1)N1CC(CCNC(CSCCC#N)=O)C1.C1(N)CCCO1 C(=O)(C(CNC(=O)C#CC1CCOC1)C(C)(C)C)NCc1c(OC)nsc1 C1(CC)CCCCC1OCC(=O)N(CCN(C(=O)C(C)(C)O)C)C(C)C C(C)(C)(C(=O)N(C)CCN(C(C1CC(C)C1)=O)C(C)C)OCC N1(C(COCCCCCC)=O)CCCC(CNC(=O)C(C(C)C)N(C)C)C1 C1(CNC(=O)C(=O)NCc2nc(-c3ccc(F)s3)no2)CCS(=O)(=O)C1 Cc1c(C(=O)NC(CO)C(=O)NCc2noc(C(N)=O)n2)cccc1O C1(C(N2CC(C(C)NC(C(CC=C)(C)O)=O)C2)=O)CN(C)CCN(C)C1 C(=O)(C(O)C1=CCCCC1)NCC1(C(N2CC[Si](C)(C)CC2)=O)CC1 CN1CCN(C(C2CC(=C3CC3)C2)=O)CC1CNC(=O)CSC1CCOC1=O C(C(CC(F)(F)F)NC(=O)Cc1ccns1)NC(CCc1nnc(C)n1C)=O c1(OC)cc(COC(=O)CCN2CCCS2(=O)=O)cc(S(C)(=O)=O)c1 N1(C(CC2(COC)CCC2)=O)CCC(NC(=O)Cc2coc(C3CC3)n2)CC1C C12(CCNC(C(C)(C)C3CC3)=O)CCC1CN(C(C1CC(F)(F)CS1)=O)C2 c1(C(N2CCC3(NC(C(C4CCCCC4)C)=O)C(C2)C3)=O)c(O)cc(F)cc1F C(C)(C(C)C(=O)NC(C)Cc1cn[nH]c1)NC(C1(CCOC)CCC1)=O C(=O)(C(F)C(C)(F)F)N1CC(CCNC(c2c(OC(C)C)n[nH]c2)=O)C(C)C1 Cc1nc(C(=O)NCC(C2CC2)NC(=O)C(C)n2cncn2)c2ccccn12 Cc1cc(C(N2CC(O)(CNC(=O)C(CO)c3ccccc3)C2)=O)nn1CCO N1(C(Cc2cn(C)nn2)=O)CCC(CCNC(C2CC(=C3CC3)C2)=O)CC1 CC(C)(CCNC(=O)CCCCC1CC1)C(=O)N1CCC(C(C)(C)C)CC1 c1(N2CCC(N(C(=O)CCn3cccn3)CCC)C2)nc2ccccc2s1 C1(CC)(OCCNC(=O)NC(C)C(C)OCC)CCOCC1 C1(C(=O)NCC2(C)CCN(C(CC3C(C)=NN(C)C3=O)=O)C2)COC2COCC12 C(CCOc1ccccc1)(C(=O)O)N(CC(=O)OC(C1CCCO1)=O)C.C(Cl)O C#CC1CN(C(=O)C(C)CN(C)C)CCN1C(c1ccc2c(c1)CCC2)=O c1(NC(C2C=CCN2C(c2nc(Cl)sc2Cl)=O)=O)nc(Br)ccc1Br c12cnc3n1CC(CC3)CC1C3(CN(C3)C2=O)C1.C1(C(F)(F)F)(CO)N=N1 c1(C2(CC#N)CC2)cn(C2CCN(C(c3ccccc3)C3CC3)C2)nn1 N1(C(c2cccc(C)c2Cl)=O)CC2CCOC2(CNC(c2c(C)noc2N)=O)C1 C(C(C)(CC(C)C)C=O)NC(Cc1cc(C)[nH]c1C)=O.c1(CNC(=O)OC)ncco1 C1(CC=C)(SC)CN(Cc2c(C(C(C3(N)CC3)=O)=O)onc2)C1.SCC Cc1c(O)cc(C(N2CCC(NCc3cc(-c4ccccn4)[nH]n3)C2)=O)cc1O CC(C)CC(Cc1ccccc1)C(=O)N(C)Cc1cn(CC2(O)CCCC2)nn1 C1(C(N(CCC(C(C)C)NC(=O)COC2CCCC2)C)=O)CCC(C2CCC2)CC1 N1(c2n(C3CC=CC3)nnn2)CCc2cccc(Cl)c2C1 N1(C(CCCOC(C)=O)=O)CCC(C(=O)N(C2CC2)CC2CCOC2C)CC1 CC(=O)CCCCC(=O)NC1CCC(C(=O)NC(c2nccs2)C)CC1 Cc1cccc(C(=O)NC2CC3(CNC(c4ccccn4)=O)CC2CO3)c1O C(=O)(CCCN(C)C)N(CCN(C(=O)COCC1CCCO1)C(C)C)C c1(OC)ccc(CNC2C3CN(C(c4cc(C)cc(Cl)c4)=O)CC23)c(Cl)c1 C1(CC)CN(C(C2CCC3(CC3)N2C(c2cc(C)cc(O)c2)=O)=O)CCCO1 Cc1c(C(N2CCN(C(=O)CN3CC(C)C3)C(CO)C2)=O)sc2cncn12 S(=O)(=O)(c1cc(-c2cnc(OC)cc2C(N)=O)c(C)cc1C)N(CCOCC)CC C=CCC(CC)C(=O)NCCC(C)N(C)C(c1ncn(C)c1Br)=O c1(NC(C=C(C)CNC(=O)CN)=O)ncc(F)cc1N C1(C(=O)NCC2CCCN(C(c3cnc(C)o3)=O)C2)CCC2C(C1)C2(F)F Cc1ccc2ncn(CC(=O)NCC3CCC(C)N(C(=O)C4=CCOC4)C3)c2c1 c1(CCC(=O)NCCSCCN2CCC2)csc(Br)c1.C1(=O)CO1 c1(OC)cc(C)c(C(=O)NC2CN(C(c3c(C)noc3N)=O)CCC2C)c(C)c1 c1(C(N(CCCNC(c2c(OC)ccnc2)=O)C2CC2)=O)cnc2[nH]ccc2n1 c1(CC(COC)O)ccc(SC)c([N+](=O)[O-])c1.N12CCCN1CC2.CC(F)(F)F C1(CCOC)(NC(c2nc(C3CC3)oc2C)=O)CCN(C(C2(Br)CC2)=O)C1 C(=O)(C(F)CC(C)(C)C)N(CC(=O)NCCC(C)O)CCC C1(C(N2CC3(CN(C(OC4CC(=O)NC4=O)=O)C3)C2)=O)CCn2cncc2C1 N1(C(CCc2ccc(C(=O)OC)cc2)=O)Cc2cccc3c2C(CCC3)C1 c1(C(=O)NC2CN(C(C=CC(CC)C)=O)CC2O)c(CC)ncnc1CC c1(C(NOC(CC#C)C)=O)cc(CNC(c2nccn2CC)=O)ccn1 C1(CNC(C(C)=CC)=O)CCCN1C(=O)C(CC)NC(=O)COC C1(CNC(CCN(C(C(COC)COC)=O)C)=O)OC(=O)CC1(C)C C1(NC(=O)COC2COC2)CCC(NC(C2CCCO2)=O)CC1 c1(C(C)C)ncc(Br)c(N2CC(NC(C3CC4CC3C3CC43)=O)CCC2C)n1 Cc1n[nH]c(C)c1CC(C)C(=O)N(C)CC1CN(C(=O)CSS(C)(=O)=O)C1 C1(C(N(CCC=C)CC)=O)CC2CC1CC2NC(C1CC1(F)F)=O N1(C(C2(C)CCCCC2N(C(c2ccnc(F)c2Cl)=O)CC)C)CC2CC(CO)C2C1 N1(CC(C)C)CC(C(=O)Nc2cccc(Cn3cc(C4CCC4)nn3)c2)CC1=O C=CC1OCCCC1C(=O)NC1CC(NC(C2Cc3nccn3C2)=O)C1 C=C(C)C1CN(C(=O)C2=CCC(NC(=O)CCC3CCCC3)C2)CCO1 C1(C(=O)NCCN(C(CC)C)C)CC2CC1CC2NC(=O)C#CC(C)(C)C CCC(C(=O)OC)C(=O)N1CC(NC(c2cc3scnc3[nH]2)=O)C(C)C1 c1(OC)nn(C)cc1CNC(=O)CC1CC(C)N(C(=O)CC(Cl)Cl)C1 C(C(CC(C)C)C(=O)NCc1c(C)ncn1C1CC1)N(C)Cc1ccc(CC)s1 C(=O)(C#CC1CC(F)(F)C1)N1CCN(C(C=CC=CCCCCC)=O)C(C)C1 c1(CC(N2CCCC(C(N3CCC(O)(CO)C3)=O)C2)=O)ccc(F)c(Cl)c1 C1(NC(C(CO)OC)=O)CS(=O)(=O)CC1NC(=O)CCSc1nnnn1C C1(CCC(=O)NCCC2CC(C(=O)NCC(C)N(C)C)C2)CCN(C)CC1 Cc1cccc(C(=O)NC2CN(C(C3(C)CSC3)=O)CC23CC3)c1F CCC(CNC(=O)CCCC#N)(CC)NC(=O)C(=O)NC1CC1 C1(C)(OC)CCCN(C(C2(C#N)CC2C(F)(F)F)=O)C1.C12CCC(CC1)C(=O)N2 Nc1cccc(F)c1C(=O)NCC1CCCCN1C(=O)Cc1cncnc1O C1(C(=O)NCCN(C(C)=O)C)CCC(C(N)=O)CC1.C12(CC1)C(=O)O2 N1(CC(=O)N(CC2(CC)CN(C(C3CC3C(=O)O)=O)C2)C2CC2)CC2C=CC1C2 C(=O)(N=c1[nH][nH]cc1C(C)(C)C)N1CC(C)N(Cc2cc(Br)cc(I)c2F)CC1 O=C(CN=c1cc[nH]cc1)NC1CCN(C(=O)CCCCF)CCC1CO c1(OC)ccc(C(N2CC(CNC(c3cncs3)=O)C3CC23)=O)c(F)c1 C1(CC)CN(CC(N2CCN(Cc3cscc3OC)CC2)=O)CCS1 C12(NC(CC3CC(=O)NC3=O)=O)CCCC1N(C(=O)CC1CCCC13CC3)CC2 n1(C(C)C(=O)NC23CC2CN(C(=O)CCCC2CC2)C3)ncc2ccccc12 c1(SC)nc(C)cc(=NCC2(O)CCN(C(C3CC3(F)F)=O)C2)[nH]1 C1(C(=O)NC(C)(C(=O)NCC(=O)N2CCCO2)C2CCC2)CCC2(CCC2)O1 C1(O)(CNC(C(C2CCC2)OC)=O)CCCN(C(=O)COc2cnc(Cl)cn2)C1 C(=O)(C=C1SCC(=O)N1C)NCC1CN(C(C(CC)SC)=O)CC12CCC2 C=CCC(Cc1ccccc1)N=c1cc[nH]c(=NCCC2=COCCO2)[nH]1 C#CC(C)(C)C(=O)N1CCOC(C(=O)NCC2(C#N)CCC2)C1 CC1CN(C(=O)CC(c2ccc(Cl)cc2)O)CCN1C(c1cnccn1)=O Cc1c([N+](=O)[O-])c(CC(C)NC(C2CCCCCN2C(=O)OC(C)(C)C)=O)nn1C c1(OC)ccsc1C(=O)NC(C1CCN(C(=O)CC(C)C)C1)C.C1(=O)CCN1.C C(=O)(C(O)C(C)C)NCCCCCCOCCN(C(C(CO)OC)=O)C C12(C(N3CC(O)(CN(C)C(C45CCC(CC4F)C5)=O)C3)=O)CC1COC2(C)C C(=O)(C(C#N)C(C)(C)C)NCC1OCCC(NC(C2CCC(C)(C)CC2)=O)C1 C=CC(C(=O)NCC1(C(=O)NC(C)C)CC1)NC(c1ccn(CC)n1)=O c1(CCC)cc(C(=O)NCC2(O)CC(NC(=O)CN3CCC(C)CC3)C2)c(C)o1 c1(C(C)NC(=O)NC(c2ncn(C)n2)C)ccnc(F)c1 C1(NC(C2(C(=O)NC)CC2)=O)COC2(C1)CN(C(c1nc(Cl)c(Cl)s1)=O)C2 Cc1nn[nH]c1C(=O)N(CCNC(=O)CCC#N)Cc1ccccc1 C(CCC(=O)NCCCOCCC(N1CCCC1CN(C)C)=O)=C(C)C N1(C(c2cc(C)c(Cl)cc2F)=O)CCN(C(=O)Cc2ccco2)C2CCCCC12 c1(C(C(=O)NCCN(CC(C)O)C(C2C(C#C)C2)=O)(F)F)ccc(C)cc1 N1(C(CCC2CCN(C(C(C=C)O)=O)CC2)=O)CCC2(CC1)CN(C)C2.C(C=C)O C1(C)(CNC(CN(CC)CC)=O)CN(C(c2oc(C(F)F)cc2C)=O)CCO1 C1(OCC(=O)NC(C)CC2CN(C(=O)CSc3nncs3)C2)CCC(F)(F)CC1 N1(CCNC(CC2CCN(C(CC)(C)C)C2)=O)c2ccccc2N(C)S1(=O)=O Cc1ccnc2sc(C(=O)N(CCCNC(C3CC(C)(O)C3)=O)C)c(C)c12 C(=O)(C1=NOC(C)C1C)NCc1ccc(CNC(Cn2c(C)nc(C)n2)=O)cc1 c1(N2CCN(Cc3c(Br)cc(CC=C)c(O)c3)CC2)ccc(I)c([N+](=O)[O-])c1 c1(C(=O)NC2C(CNC(C=CC(=O)OCC)=O)CCC2)cc(=O)c(OC)c[nH]1 Cc1cscc1Cn1cc(CC(C(=O)O)NC(=O)C(c2ccccc2)C)nn1 CCC1CCC(=O)O1.C1(C(=O)NCCC(=O)N(C)C)CN2CCN1CC2 c1(CC)c(C(=O)NCC(C)N(C)C(C2CC3(CCC3O)C2)=O)sc2ccccc12 c1(CNC(c2c(C)nns2)=O)ccc(CNC(C2(C)CCCCO2)=O)c(F)c1 c1(C(=O)NCC(CC)NC(=O)CSCCOC)csc(-c2ccoc2)n1 C1(NC(c2c(COC)cccn2)=O)CC(O)CN(C(=O)Cc2cnc[nH]2)C1 n1(CC(=O)NCC(C2CC2)NC(C(C)C#N)=O)ccc2c(=O)n(C)c(=O)n(C)c12 c1(C(=O)NCC2(C)CN(C(c3ccc[nH]3)=O)C2)ccc(NS(C)(=O)=O)cc1Cl N1(C(C)=O)CC(N=c2[nH]c(=NCC3CCCC3N(C)C)[nH]c3c2SCC3)C1 CC1CCC(C(=O)NCC(C)(C2CC2)NC(=O)C(C)NS(C)(=O)=O)C1 c1(CCC)ncc(C(C(=O)NCC2CCOC2)N(C)CC)s1 N1(C(Cc2cn(C)nc2)=O)CCN(C(c2cnccn2)=O)C(c2ccccc2)C1 N1(C(C(C)C2(O)CCC2)=O)CC(C(N2CCC(OCC3CC3)C2)=O)OC(C)C1 Cc1ccc(C(=O)NCC2CC2)c(C2CC2)c1.C1(C)CCCN1C(c1occc1Cl)=O C1(C(N(CCC)Cc2noc(C)n2)=O)CCN(C(=O)CC2CCO2)C1 C1(NC(CNC(C(CC)C)=O)=O)CCN(C(=O)CC2CCCC2O)C12CC2 N1(C(CN(C)C)=O)CCC(O)CC1C(=O)NC1(CO)CCSC1 C1(C(=O)NC2CN(C(c3c(OCC=C)cc(Cl)cc3)=O)C2)CC1C1CCOCC1 C(=O)(C(C)(C)C(C)C)NCCN(C(C1(CCC)CCC1)=O)C N1(C(c2c(CC)csc2)=O)CCC(CO)(CNC(C2(CO)CCOC2)=O)C1 N1(C(CCCCOC)=O)CC2CC1CN(C(C1CCS(=O)(=O)C1(C)C)=O)C2 NS(=O)(=O)c1coc(C(=O)NC2C3CC2CN(C(=O)Cn2nccn2)C3)c1 CCCC(CC)C(=O)NCCC1CN(C(C23CC4CC2C3C4)=O)CCO1 C1(CNC(COCc2cc(C)no2)=O)CC2CCC1N2C(c1csc(Cl)n1)=O C1(CN(C)C(c2cnc(CC(C)(C)C)o2)=O)CN(C(=O)CC2CCC2)CCO1 CCC(C)CN=c1nc(N2CCN(CCSC)CC2)c2c([nH]1)c(C)nn2C C(C(CC(C)C)NC(=O)CCC1CC1(F)F)NC(Cc1cc(C)ns1)=O C(=O)(C#CC1(CC)COC1)NC(C(=O)N(C(CC)CC)CC(C)C)c1ccco1 c1(C(N(CC(C)O)CCNC(C2CC2F)=O)=O)cc(C(N)=O)cc([N+](=O)[O-])c1 c1(C(=O)NC2(C#C)CCCC2)ccc2c(c1)N(C(=O)OC(C)(C)C)CCS2 C1(NC(C2N(CCC)CCCC2)=O)CC2(CCCCN2C(C2CCC2)=O)C1 C1(CC(=O)NC2CCN(CCF)C2)(CNC(=O)CN2CC=CC2)CCCC1 N1(C(CCSCCCC)=O)CCC(NC(=O)C(O)C2CC2)C(O)C1 Cc1cc(C(=O)NCC(C)(C)CNC(c2nccc(Cl)c2C)=O)nc(C)c1 c1(CC)ccc(C(=O)NC2CCC(C)(NC(=O)CCc3cnco3)CC2)cc1F C1(C(=O)NC2CCCC(NC(C3(C=C)CC3)=O)CC2)CC2CCC(C1)N2C CC(CC(F)F)C(=O)NC12CC(CNC(=O)CCC3CCCO3)(C1)C2 c1(C(=O)NCC2CC(OC)C2)cc(C)c(-c2ccc(CO)cc2)cn1 CC1CN2CCN1C(C(=O)NC1CC(NC(c3ccc(F)c(O)c3F)=O)C1)C2 N1(C(CC=CC=C)=O)CCCC(N(C)C(c2cc(C(N)=O)ccc2OC)=O)CC1 CC1(C)Cc2ccccc2CN1C(c1ccc(Cl)o1)C(=O)Nc1ccccc1 C(=O)(C1=NN(C)C(=O)CC1)N1CCN(C(C(CC)O)=O)C(CC2CC2)C1 c1(C(N(C2CCN(C(C3CNC(=O)C3)=O)C2)CC)=O)csc(C(F)F)c1 CCCC(CNC(=O)CCc1cncs1)NC(C12CC(C1)C2)=O C(c1ccc(C(=O)O)o1)=CC(=O)Nc1ccc(NC(=O)Oc2ccc(Cl)nn2)cc1 c1(C(N(C(COCC)C)C)=O)nc(Cl)ccc1N.C12(CCCCC1)C(=O)N2 c1(C(N2CC(C(C)NC(CCSC)=O)C2)=O)c[nH]c2cccc(C)c12 c1(CC(=O)N(C2CN(C(=O)CC3(C)CC3)CC2F)C)cncc(F)c1 CCCC1C(=O)NCc2nccc(n2)CN1.c1(N2C(CC)CCC2)ccccc1 C1(NC(CCC(=O)NC)=O)CC2CC(NC(c3cnccc3C)=O)CC12 CCCCC(O)C(C)C(=O)NC(CCC(=O)NC(C)(CC1CC1)C1CC1)C(C)C C1(C(N(CCS(C)(=O)=O)C)=O)CCN(C(C2CCS2(=O)=O)=O)CCO1 N1(C(C2C(CNC(COC3(C#C)COC3)=O)CCCC2)=O)CCc2c[nH]nc2C1 C1(NC(=O)CC2C=CC(NC(=O)C(F)=CC3CC3)C2)CNC(=O)OC1 N1(C(CC(C)C)=O)Cc2ccnn2CC(NC(=O)C(F)C(C)(C)O)C1 C1(NC(c2ccc(C(C)=O)[nH]2)=O)CN(C(c2ccc(O)cc2C)=O)CC1(C)C C(=O)(CC(C)F)N1CC(C(C(=O)NCCNS(N)(=O)=O)OC)C1 N1(C(CCCN(C(C)C)C)=O)CC(C)(C(N2CC3CCC2C(O)C3)=O)CC1(C)C c1(C(N(C)CC2CCSC2)=O)ccc(CNC(C2OCCC2(C)C)=O)nc1 C(=O)(C1=NOC(C)(C)C1)NCC1N(C(c2cc(C)c(Br)s2)=O)CC2(CC2)C1 N1(C(C(C)Cc2cnn(C)c2)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(CO)C1 c1(C(=O)NC(C2CCN(C(C3CC(=O)N(C4CC4)C3)=O)C2)C)cc(C(F)F)ccn1 c1(C(=O)NCCCN(CC(O)C(=O)NCCOC)C)cc(Cl)c(Cl)c(Cl)c1 c1(C(=O)NCC2C(NC(c3n(C)nnc3)=O)C2)csc(Cl)c1Cl c1(NC(c2c(C(=O)OC)n(C)nc2)=O)ccccc1NC(C)=O N1(C(c2cc(C(C)=O)c(C)o2)=O)CCC(NC(c2n[nH]cc2Cl)=O)C(CO)C1 c1(C(=O)NCCC#CC)cccc(CNC(C2CCCC(N(C)CC)C2)=O)c1 S(=O)(=O)(c1cccc(F)c1)NC1CC(N(C(=O)CC2CC3(COC3)C2)CCO)C1 N1(C(CCOCCC)=O)CCCC2(CCN(C(c3cc(C)n(C(F)F)n3)=O)C2)C1 c1(-c2onc(C(C)(C)C3CC3)n2)ccc(N2N=CCC2=O)c([N+](=O)[O-])c1 N1(C(C2(c3cccnc3)CC2)=O)CC2CCC(NCC3(C)CCCOC3)CC2C1 c1(CCOC)nnc(N(C(C)CNC(=O)CC2CC(F)(F)C2)C)s1 S(=O)(=O)(c1cccnc1NC1CC(=O)N(C2CC2)C1)NCC(CC)O c1(OC)cccc(C(=O)NCC(O)CCNC(C2CC2c2ccn(C)n2)=O)c1C CC(C)C(C)(O)C(=O)N1CCC(C(C)NC(c2cnnc(O)c2)=O)C1 c1(C(=O)OC(C)(C)C)cc(C(=O)NCCCCNC(C2CCCCS2)=O)[nH]n1 N1(C(CCC=CC)=O)CCN(C(=O)Cc2c[nH]c3cccnc23)C(C)C1C N1(C(C(C)(C)C2CCCO2)=O)CC2CC2(CNC(c2ccncc2F)=O)C1 CC1(C(=O)NOCC2CCOC2)C=CCN1C(C1CCSCC1)=O C1(NC(C2C(C)(C)CC2)=O)CCC2CC1CN2C(=O)C=Cc1ccc(=N)[nH]c1 C1(N(C)C(c2cnco2)=O)CCCC(N(C)C(c2ccnc(O)c2)=O)C1 c1(C(N2CCCCC(NC(=O)CCc3cscn3)C2)=O)ccc2nncn2c1 c1(C(N2C(CNC(=O)CC3CC=CCC3)CCC2)=O)cc2c(=O)cc[nH]c2s1 C(=O)(C1CCCc2scnc21)NC1C(NC(Cc2c(C)ccs2)=O)CC1 C1(n2cc(-c3onc(C)n3)nn2)CN(Cc2cc(Br)no2)CC1C CCC(C#N)C(=O)N(C1CCCCC1)CCNC(=O)C(C)(C)Cc1ccccc1 n1(CCC)cccc1C(=O)NCC(C)C(=O)NCC(=O)NCCO Cc1nc(C(N2CCC(CCNC(C3CCCCS3(=O)=O)=O)C2)=O)c(C)n1C Cc1cc(C(C(=O)N(C2CCOCC2)CCF)CC)cnc1C.c1(CN)ccccc1 C(=O)(CC(C)C(C)(C)C)N1C(NC(=O)NCc2c(C)cnn2C)CC(N=[N+]=[N-])C1 N1(C(c2ccc(C)cc2)=O)CCC(C2CCN(C(=O)C(F)CC(C)(C)C)CC2)C1 C#CC(C(C)C)NC(c1conc1C(C)NC(c1cc(CCO)on1)=O)=O c1(C(N2CC(CNC(CC3COCC(C)O3)=O)C2)=O)cc(Br)ccc1N C12(C(NOCC(N3CC(CCOC)(OC)C3)=O)=O)CC(CCO1)C2 N#CC1CN(Cc2ccc(C(F)(F)F)cn2)CCN1C(c1cccc(O)c1F)=O N1(C(C(COC)NC(=O)Cc2ncoc2C)=O)CC2(C1)OC(=O)NC2C c1(C(=O)NC(CCNC(C2CCN(C(C)=O)C2)=O)C)cc(C(F)(F)F)ccc1O Cc1c(C(=O)Nc2ccnc(OC3CCCC3)c2)[nH]c2c(Cl)cccc12 C1(CC)Cc2ccccc2CN1C(C(=O)NCCC1CC1)C1=CCSC1 N1(C(Cc2c(C)ocn2)=O)CCC2(C1)CN(C(c1cccc(F)c1Br)=O)C2 Cc1cc(=NCC2(CO)CC3CCC2CC3)[nH]c(=NCC(=O)N=S(C)(C)=O)[nH]1 C(C(=O)N=c1ccn(CC=C)[nH]1)N(C(=O)C(CCC)N(C)C)CC#C c1(NC(N2CC3(OCC(C(=O)OCC)C3)C2)=O)cnc(O)c2c1NCCC2 C1(NC(CN2CC(C)C2)=O)CC2CC1N(C(C1(C)CC=CCC1)=O)C2 c1(-c2cn(C(C)C(=O)NC3C=CCN(C4CC4)C3)nn2)cccc(C(=O)O)n1 N1(C(c2ccc(CC(C)C)nc2)=O)CC2(C1)CN(C(=O)C(F)=C1CCC1)C2 C(=O)(C(C)CC(=O)N1CCOC(C)(CNC(=O)CSCc2cccs2)C1)OC C1(C(=O)NC(C)CNC(=O)CCn2cccn2)CC12CCOc1ccccc12 C1(C(=O)NC2C(NC(=O)CCc3nncs3)CC2)CC2(COCCO2)C1 Cc1ccnc(C(=O)NC2CCCCC2CNC(=O)Cc2ccno2)c1N c1(CN2C(C(=O)NC(C3CCOCC3)C)C3CCC2C3)cc(O)c(Br)cc1O c1(C(=O)NCC2(O)CCN(C(Cc3c(C)cco3)=O)CC2)ccn2cccc2c1 c1(C(=O)NCC(CCC)NC(C2CCCC2(C)C)=O)ncncc1Cl C(C(C)(C)C(=O)NCC1CC(NC(=O)CCc2ccc[nH]2)C1(C)C)OCC c1(CC)ncc(C(N2CCC(NC(=O)C(C)OCC(F)(F)F)CC2)=O)c(O)n1 c1(OC)ccn2cc(C(N3CC(C4CN(C(C5CNC(=O)C5)=O)C4)C3)=O)nc2c1 C1(NC(c2c[nH]c(C(F)(F)F)n2)=O)CC2CN(C(c3cc[nH]n3)=O)CC2C1 C1(n2cc(C(C)OC)nn2)CCC(C(=O)NCC2CCOCC2)CC1 C1(C)(C(=O)OC)CCN1C(=O)C(CNC(=O)C(N1CCCCC1)C)OC c1(N2CCC(NC(c3c(CC)scn3)=O)C23CCC3)ccnc2nc(C)nn12 N(C(=NCCC(C)=O)NC(c1cc2ccccc2o1)C)CC(CC)n1cccn1 N(C(=NCC1CC1)NCc1cccc(Br)n1)CCCC=C(C)C Cc1ccc(S(=O)(=O)NC(c2ccc(CN3CCC4CC34)cc2)=O)cc1 C1(NC(C2NC(=O)CC(C)C2)=O)CCC2CN(C(=O)Cc3ccon3)CC2C1 c1(C(C(N2CC3C(NC(=O)C4=CCCCC4)C3C2)=O)=O)c[nH]c2cc(F)ccc12 c1(CC(=O)N(CCCNC(C2=C(C)CCC2)=O)C2CC2)ccc2c[nH]nc2c1 c1(OC)cc(C2CC2COC(=O)C(C2CCS(=O)(=O)CC2)O)ccc1F Cc1cc(C)c(C(=O)NC(C(=O)NOCC(=O)N(C)C)C2CC2)o1 C1(C(N(CCCN(C(C2(OCC)CCOC2)=O)C)C)=O)CCn2cncc2C1 c1(C(=O)NCC2CC(NC(C3C(C(C)(C)C)C3)=O)C2)ccoc1C1CC1 C1(C)(CC)CCN(C(=O)Cc2coc(-c3ccccc3)n2)C1 CC1C(CC(=O)NCCC2(O)CN(C(=O)C(C)S)C2)C1(F)F N1(C(c2nnn(C)n2)=O)CC2C3CCC(C2C1)N(C(c1cncc(N)n1)=O)C3 C1(OC)(CNC(C2CC(=C3CC3)C2)=O)CCN(C(=O)CN2CCCCC2)C1 c1(CNC(=O)NCCSC)ccn2nncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1cccn1)NCCC(=C)C Cc1nsc(C(=O)NCC2(C)CCCN2CC(C2CCCCCC2)O)c1Br c1(C(=O)NCCCOCCCNC(C(C)SCCCC)=O)c(F)ccc(F)c1O C1(C)(C(N2CC(CNC(C)=O)C2)=O)CCN(C)C1=O.N12CCN(CC1)CC2=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC(CNC(c1n(CC)c(O)nc1)=O)CCOC C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC(C)CN(C(=O)C=C1CCCCC1)C N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CC(F)CC1CNC(=O)CSC(F)(F)F C=CCC(CC)C(=O)NCc1ncoc1CCNC(=O)CC1CCOC1=O C1(C(N(C(C)CCNC(=O)CCS(N)(=O)=O)C)=O)C(C)(C)CCCC1(C)C c1(-c2ccc(F)nc2)cnn2c1CN(Cc1ccc(Br)cc1Br)CC2 CC(=O)CCCCC(=O)N1CCC2CC12C=O.N1(CC)CCC2(CCC2)CC1 N1(Cc2cc(-c3cccc(OC)c3)no2)CCC2(CC1)CC(C(=O)N(C)C)CO2 N1(C(c2c(CC)non2)=O)CCOC(CNC(=O)CC2C=CCC2)C1 C(CCCN=[N+]=[N-])COC1CCN(C(C(C)CNC(=O)CSC2CC2)=O)C1 Cc1nc2sccn2c1C(=O)NC1CC1NC(c1cnc2cnccc2c1)=O C1(NC(c2cnc(C(N)=O)s2)=O)CC2(C1)CC(NC(c1ccc(F)cc1N)=O)C2 N1(C(CCSCC)=O)C2CCC1CC(N(C)C(C1CCCN(C(=O)CC)C1)=O)C2 c1(C(C)=O)ccc(C(=O)NCC2CCN(C(c3ccc(F)cn3)=O)CC2)cc1O C1(C(=O)NC(C=CC(=O)N(C2(OC)CC2)CC)C)CCCC1C C1(NC(C(C)c2cccs2)=O)CCCC(C(=O)NC2CN(C)NC2=O)C1 C1(C)(NC(c2cc(C)sc2Br)=O)CCCN(C(C2(c3ccno3)CC2)=O)C1 N#Cc1cccc(CC(N2CCCOC(CCNC(c3ccsn3)=O)C2)=O)c1 c1(C(CC)NC(=O)C(CC2CCCCC2)CC)cccc(S(=O)(=O)N(C)C)c1 N1(C(C(C=C)O)=O)CC(F)(F)CC1CC(=O)NCc1ccncc1F c1(C(=O)NCC(C)N(C)C(C2CCC3CCC2O3)=O)nn(C)c(Cl)c1Br N1(C(C(C)SCC)=O)CCN(C(=O)CCC(=O)c2cnn(C)c2)C(CO)C1 n1(C(=O)NC2CN(C(=O)COCCF)CC23CC3)ccc(=O)c([N+](=O)[O-])c1 C1(CCOC)C(=O)NCCN1C(=O)C(N)CCc1cccc(C)c1 c1(C(=O)NC2CC(C)(C(=O)NCc3cc(C)c(F)cc3)C2)cc(F)c(N)cc1F Cc1cc(=NC2CC2c2ccnn2C)[nH]c(NCC2CC2c2ccc(Cl)cc2)n1 C1(CCC)(NC(=O)C(F)C2CC2)CCN(C(c2snnc2C)=O)CC1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CCN(C(c3n[nH]c4c3CC3CC43)=O)CC2)C1 Cc1cc(C(=O)N(C(C)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)C)C)ccc1F N1(c2ncc(CCC)cn2)C2CCC1CC(CNC(=O)C1=CS(=O)CCC1)C2 C1(C(=O)NC2(C#N)CC2)(CNC(C(C)=C(C)C)=O)CCCCC1 C1(c2nc(SC)nn2C2CCOC2)CN(Cc2ccccc2)C2(CCC2)C1 Cc1ccc2c(c1)C(C(=O)N1CCN(C(=O)C(C)(F)F)CC1)CC2 C=CCC(C(=O)NC(C)CNC(c1ccc(CCCCC)o1)=O)N(C)C C(=O)(C1=NN(C(C)C)C(=O)CC1)NCCC(CCNC(c1c(C)cc(F)s1)=O)C C1(CNC(c2cnc(Cl)cc2Cl)=O)CCCN(C(=O)CCc2cnoc2)CC1 N1(C(c2c(C)n(Cc3ccccc3)nc2)=O)CCc2cc(C#N)ccc21 c1(OC)ccc(C(N2CCC(NC(c3cc4c(s3)CCOC4)=O)C2)=O)c(N)c1F c1(C(N2CC(CNC(Cc3cnc(C)o3)=O)C(O)C2)=O)c(C)nc(C)n1O C(=O)(CC(O)CNC(C1(N(C)C)CCOCC1)=O)NC(c1nc(C)[nH]n1)C c1(C(N2CC(N(C(=O)C(F)(F)c3cscn3)C)C(F)C2)=O)ccc(CC#N)cc1 c1(OC(CC(CC)CCOc2nc(C(C)C)ns2)C)ccc2c(c1)CCC2 N12CC3CC1C3C(=O)NC1CC(C1)C2=O.c1(OC)ccnc(C2CC2)c1 C1(C(=O)NCc2ccoc2)(NC(C(C)c2ccco2)=O)CCC(C)(C)C1 C1(C(=O)NC(CNC(C(c2cccc(Cl)c2)CC)=O)(C)CO)CN2CCC1CC2 c1(C(=O)NCCN(C(c2nc(COC)oc2)=O)C)ccc(O)c(N)n1 C1(NC(=O)C=C2CCSCC2)CCOCC1C(N(CC(O)C1CCC1)C)=O c1(C(N2C(C(N3CCN(C(N(C)C)=O)CC3)=O)CC3CC32)=O)nccc2nc[nH]c12 C1(NC(CC(n2c(CC)ncc2)C)=O)CC(C)CN(C(=O)CN2CC(C)(C)C2)C1 Cc1cc(C(N)=O)ccc1CNCc1cc(Br)c[nH]1 Cc1cc(CC(N2CC(O)(CN(C)C(c3ccc(C)nn3)=O)C2)=O)cc(C)c1 N1(C(=O)C2=CCCS2)CCCCCC(NC(=O)C(F)(F)c2ncccn2)C1 c1(NCC(CC)S(N)(=O)=O)ccc2c(O)cc(OC)nc2n1 C1(N(C)C(c2cccc(=O)o2)=O)CN(C(=O)CC2CCS(=O)(=O)CC2)CC12CC2 C1(CNC(c2n(C(C)C)ncc2)=O)C2CC1N(C(C1CCSC1)=O)C2 Cc1cc(C(N2CC(C)(CC(N3CCC4(CC4)C3)=O)C2)=O)nc(C)c1 c1(OC)ccc(S(=O)(=O)NC2CC2)cc1CC(=O)O.C12CC1OC2 N1(C(C=CC=CCC)=O)CC2CCC1C1CN(C(=O)C(F)(F)c3cscn3)CC21 C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C(CNC(c2ccc(C)c(O)n2)=O)CC1 C1(NC(C2C(CC)C2)=O)CCCC12CN(C(c1ccc(-n3ccnc3)nn1)=O)C2 C(CC(C)C(=O)NCCNC(c1ncoc1CCC(F)(F)F)=O)OC C(=O)(C(CC#CC)NC(=O)CC(CC)C1CC1)N(CCCCCC=C)C C1(O)(CNC(C2(Cl)C(C)(C)C2)=O)CCCN(C(C2CN(S(N)(=O)=O)C2)=O)CC1 C#Cc1ccc(CC(=O)N(C2CCCC(NC(=O)CS(=O)(=O)N(C)C)C2)C)cc1 Cc1ccnn1CC(=O)NCCOCCCNC(c1csc(-c2ccco2)n1)=O Nc1c(C(N2CCC(NC(=O)CC34CCCC3C4)C(O)C2)=O)cc(F)c(F)c1F CCCCC(=O)NC1COCC1CNC(c1ccnn1CC1CC1)=O C1(NC(C(C2CCCC2)NC(=O)CSC2CC2)=O)CC(O)C12CCC2 N1(C(C2C(C)(C)C2(C)C)=O)CC(NC(c2ccccc2Cl)=O)C(F)(F)C1 Cc1cc(C(=O)NCC2(O)CCN(C(C3COC(=O)N3)=O)CC2)c(C)c(C)c1 C12(NC(c3ccc(CC)cc3N)=O)CCCC1CN(C(=O)C(C)(C)C1CCC1)C2 C1(C(=O)NCCC(COC)OC)CC2C=CC1N(C(=O)CCCCC(C)C)C2 c1(C(=O)NC2CC(CNC(c3c(COC)scc3)=O)C2)coc2c1CCCC2 CC(O)CCCCCC(=O)NCC1CCN1C(C1(c2ccccc2)CCOC1)=O CCC(CC(=O)NC1CCC(NC(=O)C(c2ccc(OC)cc2)=O)C1)C(F)F c1(SC(C)C(=O)N(C2CCN(C(=O)COCc3ccncc3)C2)C)ccccn1 C(=O)(CCCCC(=O)N1CC2CC(NC(=O)C=Cc3ccc(C)cc3)C1C2)OC c1(C(=O)NCC2(O)CC(NC(CC(C)(F)F)=O)C2)cccc2c1NC(=O)CC2 C=CC1(C(=O)OCc2c(C(N(CC=C)CC)=O)cccn2)CCCCC1.N(C)C c1(NC(CC(CNC(C(CCC)CC)=O)C)=O)ccc2cnccc2c1 C1(C(N2CCCN(C(c3cnc(C(C)=O)s3)=O)CC2)=O)CCc2ncnn2C1 c1(NC(C)=O)sc(Cl)cc1C(=O)NCCNC(=O)NC1(c2ccc(C)cc2)CC1 N1(C(=O)CS)CC(C(N(CCC#C)CC)=O)C1.C1(C(=O)NCCOC)CCC1 C1(C)(C(N2CC(CC)N(C)CC2)=O)CC(O)CN1C(=O)Cn1cc(C2CC2)nn1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(CN(C(CCC)=O)CC)CC(NC(C)=O)C1 C(=O)(C1=CC2(CCOCC2)C1)NCC(CNC(C1CCCC(C)C1)=O)CO C1(CNC(=O)C=CC2CCC2)CCN(C(C2CCCN2C2CC2)=O)CC1(F)F C1(NC(C(C2CN(C(c3ncoc3C)=O)C2)OC)=O)CCN(OC)CC1 Cc1cccc(CN2C(CCNC(C3CCCC(C(N)=O)C3)=O)CCCC2)c1 N1(C(C)C)CCC(NCC(C2CC2)Nc2cc(O)ncn2)CC1.C1CC(=O)N1 N1(C(c2nccc(C)n2)=O)CC2CCCCC2(CNC(=O)CC=CCN(C)C)C1 N1(C(C2C(C=C)CC2)=O)CC(NC(=O)COCc2ccncc2)CC2(CC2)C1 C1(C)(NC(c2c(C(C)C)n[nH]c2)=O)CCCCC1C(=O)NCCCC1(O)CCC1 C1(C)(CN(C(C=CC)=O)C)CCN(C(=O)CCCCNC(=O)OC(C)(C)C)CC1 N1(C(C(C)OCCOC)=O)CCOC(C)(CNC(C2(C)CCC3CC3C2)=O)C1 N(C1CN(C(=O)Cc2occc2C)Cc2ccccc21)C(Cc1nc(C)sc1)=O CC1(C)CC(CNC(=O)CS(N)(=O)=O)CN(C(c2cnc(O)c(Cl)c2)=O)C1 CCC(C(=O)NC1CCC(CNC(c2ccc(C)nn2)=O)C1)C(F)(F)F C1(NC(C(=O)NCC2(C)CCOCC2)=O)CCCC[Si](C)(C)C1 C1(NC(C=C(CCC)C)=O)(CO)CCN(C2CCN(C3CCCC3)C2=O)CC1 N1(C(C(C)n2cccc2)=O)CCC2(CNC(C3(CCF)CCC3)=O)CCCC12 N1(C(c2c(C)ccnc2O)=O)CCCN(C(=O)CCOC2CCCCC2)CCC1 N1(C(c2c(C)cc(=N)[nH]c2)=O)CCCc2c(-c3nn[nH]n3)cccc21 c1(N(C2CCN(C(c3cc(C4CCOCC4)no3)=O)C2)C)ncnc(Cl)c1F C1(C(=O)Nc2ccc(SC3CC3)cc2)Cc2c(Br)cccc2CN1 CC(C)C#CC(=O)N(C(C)CNC(c1ccc(-c2ncon2)cc1)=O)C CCCC(C)(CCC)C(=O)OC.N12CC3CCC(C1)N3C(=O)CCCCC2=O c1(CN(C2CN(C(c3ccc(O)cc3)=O)C2)C)cc(OC(F)(F)F)ccc1O c1(C(=O)NC2C(C(=O)NC(C(=O)OC)CO)C2(C)C)cccc(F)c1 CC(C)C(C)(C)C(=O)N1CCOCC(C(=O)NC(c2nccc(O)n2)C)C1 C(c1c2c(nn1C)CCCC2)=CC(=O)NC1C2CN(C(CC(C=C)(C)C)=O)CC21 c1(COC)nc(OC)cc(NC(C2CCCC2)CNC(=O)CC(C)O)n1 c1(C(=O)NCC2CCN2C(=O)CCc2ncc[nH]2)cc2c(Br)coc2cn1 N(C1COc2cc(Br)ccc21)C(c1n(CCC)nnn1)C(C)(C)n1cncn1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC1=CCCCC1)NCCC(C(C)C)CO c1(N)ccc2c(c1)OC(F)(F)O2.ClC1(Cl)CC1CCCC1CCC1 C1(NC(C(CC)SC)=O)CN(C(=O)Cc2nc[nH]n2)CCC12CCOCC2 C1(C(=O)NCC#CC(=O)NCc2noc(C3CC3)n2)(OC)CCC(C)C1 c1(C(=O)NCC2(CNC(C(C3CC3)OCC)=O)CC2(F)F)cncc(F)c1Cl c1(C(N2CCC(C(=O)NC3COCCC3N(C)C)(CC)C2)=O)ccnc(C)c1C C1(OC(c2csc(-c3cccnc3)n2)=O)CCCC2CCOC12 C1(NC(c2c(C)ccnc2)=O)CCN(c2ccc(C(F)(F)F)cn2)CC1F C=C1CCN(C(c2c[nH]c(=NC)o2)=O)C(C(=O)NCC(C)CC)C1 N1(C(CCC#CC)=O)CC2(CCC2NC(c2nc(C)ncc2Cl)=O)C1 CCCCC(C(=O)N(C)CCN(C)C(C1CC2CC2(CCC)C1)=O)C(C)C Cc1ccc(C(=O)NC23CC2CN(C(=O)COCc2ccccc2C)C3)c(O)n1 C(=O)(C1=C(C2CCOC2)N(CCC#N)C(=O)NC1c1cc(Cl)cc(Br)c1)OC c1(C(N2CC(N(C(=O)Cn3nccn3)C)C2)=O)c[nH]c2ncccc12 CCC(C(=O)N1CC(O)(CNC(=O)CSC2CCOC2=O)C1)C(F)(F)F N1(C(C(C)n2cccn2)=O)CCC(C)(C)CC1C(=O)NCC1(C)CCC(O)CC1 C1(NC(C2(F)C(C)C2)=O)CN(C(c2onc3c2CCCC3)=O)C2(CCC2)C1 C=CC1(C(=O)NC2CC3(C2)CC3C(N2CCC(C)(O)CC2)=O)CCOCC1 c1(OC)nc(Cl)c(C(=O)NCC(C)(C)CNC(=O)Cc2nncn2C)s1 c1(C(N2CCC(NC(C(CC)N(C)C)=O)C(C)C2)=O)csc2c(OC)cccc12 N1(C(C(C2CCOCC2)OC)=O)CCN(C(c2cnn(C)c2Cl)=O)C(C(C)C)C1 c1(CCC)ccc(C(C(=O)NC(C)C)N(C2CC2)Cc2ccccc2)cc1 c1(C(N2C(C)(CNC(=O)CC(F)(F)Cl)CCC2)=O)cnc(O)c2ccccc12 c1(C(=O)NCC2(O)CN(C(=O)CCCC3CC3)C2)ccc(F)c2cccnc12 C(C(O)CC(=O)N1CCCC1CNC(=O)CC1CC12CC2)N(C)C C(=O)(CC(C1CC1)NC(=O)CCCN(C)C)N(CC(=C)C)C CC(CC(N)=O)C(=O)NCCCC1COCCN1C(=O)CCC1(C)CC1(F)F c1(C(C)C)ccc(C(=O)N(C2C3CN(C(c4ccc(=N)[nH]c4)=O)CC23)C)cc1Cl N1(C(C23CC(NC(c4[nH]cc(C)c4C)=O)C(OC2)C3)=O)CCC2CCCC2CC1 C(C(COC)CC(=O)N1CC(C(C)NC(=O)CC2CCCC(C3CC3)O2)C1)OC C(=O)(C1CCc2scnc21)N1CC(CNC(=O)COC2CCCOC2)CC(C)C1 C1(NC(CC(C)c2ccccc2)=O)CC2CC(NC(=O)Cc3ccco3)C2C1 Cc1ccc(Oc2ccc(-c3cc(C(=O)NC4(C)CCCC4)on3)cc2)cc1 N1(c2nnc(C)o2)CCN(C(c2cccc(Cc3nncn3C)c2)=O)CC1COC C(C(C(=O)NCC(O)CN(C(=O)CCC(=O)NC1CC1)C)C(C)(C)C)OCC=C c1(C(=O)NC(CN(C(c2c[nH]cc2Br)=O)CC)C)cccc2c1C(C#N)C2 C(CCCCCNC(C1(F)C2CCCC12)=O)NC(C1(CC(C)C)CCCC1)=O c1(CC)nc(C)c(C(=O)NC2CC(n3cc(-c4cccc(F)c4)nn3)C2)o1 c1(NC(N2CCCC(n3ncc(C)c3C(F)F)C2)=O)nc2ccccc2s1 CCC(C)(C)CC(=O)N(C1CN(C(c2nc(Br)c(C)s2)=O)CC1O)C C1(CC)CCOC1C(=O)NCC1CC(F)(CNC(=O)CSc2cccs2)C1 CCCC(C(=O)NCCCCN(C)C1CC1)NC(c1sccc1C#N)=O c1(C(N2CC(CNC(c3c(OC)c[nH]n3)=O)C(C)C2)=O)cc(Br)ccc1C CC1CN(C(=O)Nc2cccc(N)c2)CC1(C)C(F)(F)F c1(CC(=O)NC2(CNC(C(=Cc3cccs3)C)=O)CCC2)ccc(C)cn1 C=CCCN=C(NCC)NC(C)CC.N1(N2CCC(C)C2)CCN(CC)CC1 N1(C(C2C(C)(CC)C2)=O)CCC(O)(c2cn(-c3c(F)cccc3F)nn2)CC1 c1(N2CCC(N(C(=O)Cn3nnnc3C)CCC)CC2)nc(CC)cc(Cl)n1 C1(C(N(CCC)CCNC(=O)C(O)C(F)(F)F)=O)CC(c2ccccn2)=NO1 c1(NC(=O)N(C2CSCCC2=O)CCc2ccccc2)cccc(F)c1 N1(C(C2C(C)(C)NC(=O)C2)=O)CCC(C2(NC(c3cc(=O)cc(Cl)[nH]3)=O)CC2)C1 CC1CCn2c(C(=O)NON3CCCC3CNC(=O)C(O)C(C)(C)C)cnc2C1 C1(C(N2CC(O)(CN(C(C)=O)C)C2)=O)Cc2ccc(F)cc2O1 N1(C(C2CC(C#N)C2)=O)CC2C(CNC(c3cccc(Br)c3)=O)C2C1 N1(C(CC2(NC(C(CC)n3ccnc3)=O)CC2)=O)CCS(=N)(=O)CC1 c1(OC)ncccc1NC(=O)C=CC(C)NC(c1ocnc1C)=O c1(C(N(CC(CN(C(Cn2c(C)cnc2)=O)C)O)C)=O)c(F)cncc1Cl C=CC(C)(O)CC(=O)N(CCCCC(=O)NC(C)C(=O)OC)C N1(S(=O)(=O)c2cccc(Br)c2)CCc2ccc(F)c(F)c2C1 N1(C(C=C(C)Cl)=O)CCN(C(C2CN3CCN2CC3C)=O)CC(O)C1 C1(C(=O)NC(CCOCC)C(=O)NC2CCN(CCF)C2)CC2CC(=O)C1O2 CCC(C)(CO)C(=O)NCC1CC(O)CN1C(c1nn(C)cc1Cl)=O n1(CC=C)c(N2CCN(CCC#N)CC2)nnc1C1CCCS1 C1(NC)CCCN(C(=O)C(=O)NCC2CCN(C(=O)COC(F)F)C2)C1 C(=O)(C(CC(C)C)NC)NCc1snc(CC)n1.C123CC(C1)(C2)C(=O)N3 c1(C(=O)NC(C(C)NC(=O)COCc2ccccc2)C)cnc2c(ccn2C)c1 c1(C(=O)NC(C2CCCC2)CNC(C2(C)CC3CC3C2)=O)csc2cccnc12 C1(OC)(CNC(=O)CC2CC3(CC3)CO2)CCN(C(=O)C(C(C)C)N(C)C)CC1 C(CC)(C(=O)NC(C)CN(C)C(c1cnsc1C)=O)=CCCC C(=O)(C1CCCn2ccnc21)NC(CC)CNC(C1CC(=O)N(C)C1)=O Cc1ccc(C(=O)N(C2CCCN(C(=O)COC3CCC3)C2)C)nc1 C(=O)(C(C)(C)CCNC(=O)Cc1cccs1)NC(CCC)C(=O)NC N1(C(CCC2C(C)C2)=O)CC2CCC(C1)C(NC(C1CC1C1CCC1)=O)C2 C1(CCCC)CCN(C(C2CC(N(C(=O)CCc3ncnn3C)C)C2)=O)C1 N1(C(c2nc(CCCC)sc2)=O)CCCC2(NC(c3nc[nH]n3)=O)CC2C1 C1(NC(c2c(CC)cno2)=O)COCCN(C(=O)C(C)(C(C)C)NC(C)=O)C1 Cc1cccc(CNC(C2CC(O)CN2C(c2cccc(Cl)c2C)=O)=O)c1C c1(C(N(CCNC(=O)C=Cc2nccs2)CC)=O)ccc(C)c(C)c1N c1(CNC2(CC(=O)OC)CCCC2)c(-c2ccc(C)o2)coc1C C1(NC(C2CN3CCC2CC3)=O)CN(C(C2CC(F)C(=O)N2)=O)CCC1CO N1(C(C2C(CC)C2)=O)CC2(CC(C(=O)N(CC)Cc3ccsc3)CO2)C1 C1(C(=O)NCC(C#C)CC2CC2)C(O)CCN1C(=O)CC1CCOC1C N1(C(C(C)(C)OC(C)C)=O)CCOCC(C)(CNC(=O)CC(C)O)C1 CC1CN(C)CCC1N=c1nc2sccc2c(NCC2CCC(S(C)(=O)=O)CC2)[nH]1 Cc1nn2ccccc2c1C(N1CCCC(NC(=O)CC2CC(F)C2)C1)=O C12CC3CC1N(C3)C(=O)CC1CN2C1.c1(C(C2(O)CCC2)C)noc(CNC)n1 N1(c2ccnc(C(=O)OC)n2)CCCC(C2CC2NC(=O)C(C)(C)CSC)C1 c1(-n2c(-n3nccc3C)nc(CCC)n2)ccc(CSC)cc1C N(C1CN(C(=O)C(C)CCCOC)Cc2ccccc21)C(C=CC)=O C=C=C(C)CC(=O)NCC1(C)CCCN1C(c1cnn(CC(F)F)n1)=O N1(CCC(=O)NC(C(C)NC(COCCCCC)=O)CO)CCCCC1=O c1(C(N2CCC(C(C)NC(CCCc3c(C)ccs3)=O)C2)=O)cccc(C)c1N C1(C)(C(=O)NC(C2N(C(C(C)OCC)=O)CCC2)C)CCC(=O)N1 C(c1cc(OC)c(OC)cc1OC)=NC(CCN(CC)Cc1cccc(Cl)c1)=O N1(C(C(C)C)=O)CCC2CCN(C(c3ccc4cnoc4c3)=O)CC2C1 CC1(C)C(NC(C2CCCC2(F)F)=O)CCN1C(=O)Cc1cccc(C(F)F)c1 c1(CC)ncc(C(N2CCC2C(=O)NC(CO)C2(C)CC2)=O)o1 N1(C(c2n(C)ncn2)=O)CCC2CCN(C(c3ccn4c3CSCC4)=O)CC2C1 c1(C(=O)NC2C(NC(C(c3c(C)nn(C)c3)C)=O)CCC2)cncc2c1CCC2 C1(C(=O)NC2CCCCN(C(c3ccc(CC)nc3)=O)C2)CCCCCS1(=O)=O n1(CC(=O)NCC2CCN(C(C(C3CCCCC3)OC)=O)C2)nc(C)c(C)c1C Cc1cc(C(N2CCCC2C(C)NC(c2snnc2C)=O)=O)cc(Cl)c1 c1(C(N2CC(N(C)C(c3ccc(Cl)[nH]3)=O)C(F)C2)=O)ncnc2c1CCCC2 CC(C)(C)CCC(F)C(=O)NCC1CN(C(=O)Cc2ccc(F)cc2F)CC1O c1(OC)ccc(C(=O)NCCCc2ccc(Cl)cc2Cl)cc1-c1cccc(F)c1 C1(C(=O)NC(C)Cn2cccn2)(CNC(=O)CC2CCC2)CCCO1 N1(C(C(CCC2CCC2)NC(C2C(=C)C2)=O)=O)CCCCC(CO)C1 c1(C(=O)ON2C(c3nnc(CC)o3)CSCC2)cn(C2CC2)c2ccccc12 C(C)(C(=O)N1CC2C(CN(C(=O)C(=O)C3CCCC3)C)C2C1)(C(C)C)OC C1(CC(C)NC(c2c[nH]nc2C(C)(F)F)=O)CCN(C(C2CC2C(N)=O)=O)CC1 C12(CCNC(Cn3ncn(C)c3=O)=O)CCC(C1)N(C(=O)CN1CCOCC1)C2 C(=O)(C1CCCn2nccc21)N1C(C)CC(NC(=O)CC2(O)CCOC2)CC1 CC1(CO)CN(C(C2COCCN2C(c2cc(Br)c(F)cc2Br)=O)=O)CCC1O c1(C(=O)NC2(COC)CCN(C(c3cncn3C)=O)C2)cc2cccc(C)c2o1 C1(NC(C2CC(C)OCC2)=O)CCN(c2ncc(-c3ccccc3)cn2)CC1O N1(C(c2ncc(CC)nc2)=O)CCN(C(C2CC2CC)=O)C2(CC2)C1 C1(C2(C(N(CCO)CC)=O)CC2)CCCN1C(=O)CC1(C)CCCO1 c1(C(=O)NCCCNC(C2(COC)C=CCC2)=O)cc(C)cc(Cl)c1 C1(C(=O)NCCNC(CCCC(=C)C)=O)C2Cc3cc(Cl)ccc3C12 c1(OC)ccc(NC(C2CCC(C)N2C(=O)C(F)(F)Sc2ccccc2)=O)cn1 CCCC(CC)CC(=O)N(CC(O)CNC(c1cc(C(C)=O)cn1C)=O)C CC(F)(F)CCC(=O)NCC(F)CNC(=O)Cn1cc(F)ccc1=O C1(NC(CC2C=NN(C)C2=O)=O)CCCC(C(=O)NC2CCCC(O)C2O)CC1 C(=O)(C(CCNC(=O)Cc1ccc(-c2ccccc2)cc1)c1ccccc1)OC CC1C(=O)NCCN1C(c1ccc(CNC(C2OCCC2(C)C)=O)o1)=O c1(C(=O)NCCN(C(C(Br)=C(C)C)=O)C)cc2c(C)c(C)ccc2[nH]1 C1(CNC(CCCOCCC)=O)CC(F)(F)CN1C(=O)CCN1CCC(F)C1 Cc1ccc2c(c1)C(CC(=O)NCCN(C(c1ccoc1C)=O)C1CC1)C(=O)N2 C1(NC(C=C(COC)C)=O)CCCCC12CCN(C(c1c(OC)cccc1Cl)=O)C2 c1(OC)cncnc1C(=O)NC1CC(C(=O)NCCC=C(C)C)C1(C)C C(CNC(c1cn(C2CC2)nn1)=O)(C(C)C(C)C)NC(C1(OC)CC1)=O C(C(=O)NCCOCC)(C(C)C1CC1)N(C(c1ccc(F)cc1)C)CC N1(C(c2c[nH]c(=NC)o2)=O)CC(O)CC1(C)C(=O)NC(c1ccccc1F)C C(=O)(C1=NOCC1)NC(C)C(c1ccccc1)NC(=O)COCc1ccccc1 C1(C(=O)NCCN(CC(C)O)C(c2cc(C)sc2)=O)CCOC1(C)C c1(CCC(=O)NCC(C)(C2CCC2)NC(=O)CC(C)C)ncsc1C(=O)OC C(=O)(N=c1cc[nH]c2ccccc12)NCc1c(S(=O)(=O)NC)ccs1 c1(C(N(c2c(C(C)=O)cccn2)C)=O)cc2c(s1)C(C)(C)CCC2 C1(C(=O)NCC2CCCCC2)CN(C(c2ccc(F)c(F)c2Br)=O)CCC1(F)F C12(C(=O)OC)CCC(C(=O)OC)(CC1)OC2.C123CC(C1)(C2(C)OC)COC3=O c1(NCCCNC)nc(NCCCC(C)SC)nc2c1ncn2C C1(C(=O)NC2CCC(CC(=O)NCC(CO)N(C)C)C2)CC(C)(C)CCO1 N1(C(c2ccc(CCCC#N)cc2)C(=O)NCCCSC)CCCN(C)CC1 Cc1cc(C(=O)NC2CN(C(c3ccc(NC=O)cc3)=O)C3CC23)cc(Cl)c1 C(=O)(CC1=CCN(C)CC1)N1CCC(C(F)F)(CNC(c2nc(C)oc2)=O)C1 C1(C(=O)OC)CC2C(CC1C(=O)NCc1ccc(O)c(C)c1)C2(F)F C(C(C(=O)N(C1CCCN(C)C1)C)C(C)(C)C)NC(C(CN(C)C)O)=O N1(C(C2C(OC)(OC)CC2)=O)CCC(O)(C(=O)N(C)CCc2ccccc2)CC1 CCCC(CC(C)C)C(=O)NC(CNC(=O)CC1CCC(C)(C)CC1)CC(C)C C1(C(=O)NC(CC)C(F)(F)F)COC2(C1)CN(C(=O)C(=O)NC1CC1)C2 N1(C(C=C(C)CNC(=O)COC(C)C)=O)CCC(CCCO)C1 N1(C(C(CCC)OC)=O)CCCC12CCCN(C(c1c[nH]cc1CC)=O)C2 c1(C(N2CCC(CNC(C#CC(=O)OC)=O)C2)=O)cc2ccc(OC)cc2nn1 c1(C(=O)NC(C)C)cccc(CN=C(NCC(F)F)NC2CCOC2)c1 c1(-c2nc(NC(=O)NC3CC3)sc2)cccc(Nc2ccccc2)c1 C1(NC(CC(COC)NC(=O)CC2CCSCC2)=O)CCN(C)C(=O)C1 C1(C(C)C)CC(OC2CC(C(=O)NCCC(=O)CCOC3COC3)C2)C1 C(=O)(C1CCc2scnc21)N1CC(OCCNC(C2N(C)CC3(CC3)C2)=O)C1 C(C(=O)NOCC(O)CO)(C1C(C)CC1)NC(C1(F)CCOCC1)=O C1(C)(CNC(C(SC)SC)=O)CN(C(c2ccn(C(C)C)c2C)=O)CCO1 Cc1[nH]c(C#N)cc1C(N1CCC(OCC(=O)N(C(C)CCN(C)C)C)C1)=O c1(-c2c(CN(C)Cc3ccc(OC)nn3)n(C)nc2)ccc(OC)c(C)c1 S(=O)(=O)(c1cccc(N2CC3CC(F)CC3C2)n1)NCc1nn(C)c(O)c1 CC1=CC(C(N2CCC2CC(=O)NCC=CBr)=O)SC1 Cc1cc(N2CCC(NC(=O)CS(=O)(=O)C(C)(C)C)C(F)C2)nc(S(C)(=O)=O)n1 c1(C(=O)C=O)cn(C)nc1-c1nccs1.C(CC1CC1)(C(=O)NCC(C)(O)CN)OC N1(C(C(Cc2ccco2)NC(=O)Cc2ccsn2)=O)CCC(F)(F)C(O)C1 CC1CN(C(=O)CCCNC(C2CC2CCN(C)C)=O)CCS1=O n1(CC(N2C(CCNC(=O)CC3(CO)CC3)COCC2)=O)ccc([N+](=O)[O-])n1 c1(C(=O)NCC2(F)CCN(C(C(CC)CC(F)F)=O)C2)nsc2ccc(C)cc12 Cc1nnc2n1CCC(C(=O)NCC1(C)CCCN1C(C1CC3(CC3)CO1)=O)C2 c1(C(=O)NC(C(C)(C)NC(CC(COC)(C)C)=O)C)cc2c(o1)CCCNC2=O C(C)(N=c1ccnc(N2CCC(SC(F)F)C2)[nH]1)c1ncc(C)s1 c1(C(N2CCN(C(=O)C#CC3CC3)C(C(F)F)C2)=O)cnc2sccn12 C1(NC(C(C)C2CC2)=O)CCOC(C(=O)NCC(N)=O)C1 c1(C(=O)NCCCN(C)C(c2csc(C(F)F)n2)=O)cncn(C)c1=O C1(NC(C=CC)=O)C(C)CCN(c2ncnc(Cl)c2C)C1C CCC(C)CCCC(=O)N1CCSCC1C(N1CCC(F)(C#N)C1)=O CC1(CNC(=O)C(C)(C)c2ccccn2)CC(NC(=O)CNS(N)(=O)=O)C1 N1(Cc2cn(CC3CC(NC(c4cc(CSC)cs4)=O)C3)nn2)CCS(=O)CC1 S(=O)(=O)(c1cncc(C#N)c1)NCC(=O)NC(CCCC(C)C)c1ccccc1 C1(NC(CCc2cc(C)nc(C)c2)=O)CC12CCN(C(c1csc(O)n1)=O)CC2 c1(C(=O)NCCC(C)N(C(=O)C(C)CCN(C)C)C)cnc(O)c2cccnc12 N1(C(C(C2(O)CN(C(CC(CC)SC)=O)C2)F)=O)CC(=O)NCC1CC C12(CN(CCc3nccs3)CC)COC(C(F)(F)F)(C1)C2 C1(CCC)CN(C(=O)CCOCc2ccc(F)c(Cl)c2)CCN1C(=O)CC c1(C(=O)NC2CN(Cc3nccnc3Cl)CC2F)c(Br)ccc(Cl)c1F C12(C(=O)NCC3CC[Si](C)(C)C3)CC(CCO1)N(C(=O)CC1CCC(=O)NC1)C2 Cc1nc2ccccn2c1NC(C1(O)CCN(c2ncnc3ccccc23)C1)=O CCCCC(C(=O)NC1CC2(C1)CC(C(=O)Nc1c(O)cccc1Br)C2)NC N1(CC(=O)NCC2CCC(C(=O)NC3CCCCC3CO)C2)C(=O)CNC1=O CC(C)(C)CCCC(=O)N1CCC(Cn2cc(-c3cnccn3)nn2)C1 CC1(NC(c2c[nH]c(Br)c2)=O)CCCN(C(c2cnc(C3CCC3)nc2O)=O)C1 c1(CNC(CN2CCN(S(CC=C)(=O)=O)CC2)=O)cc(C)c(CN(C)C)cc1C c1(C(=O)NC(c2ccc(-c3cnc(C)s3)cc2)C)ccc(F)c(C(C)(C)F)c1 C1(C(=O)NCC2CCC(=O)N2)CC2CCC(C1)N2C(=O)C#CC1CCCC1 Nc1cc(C(=O)NC2CC(NC(C3C4CCC3CC4)=O)C23CCC3)cc(F)c1 c1(CN(C)C(c2sccc2C#N)=O)ccc2cc[nH]c2c1.C12CCCN(C1)C2=O Cc1cc2cc(NC(C34COCC3C4(F)F)=O)ccc2o1 S(=O)(=O)(c1ccc(NC2CC2F)c(F)c1)NCC1CC(C)CC(C)C1 c1(OC)cc(Br)ccc1C(=O)C(=O)NCC1CN(C(=O)CCC2CCC2)C1 Cc1cc(C(=O)NC2(CCNC(C3C4CC5C(C4)C35)=O)CCC2)sc1C c1(CC(=O)NC2(CC=C)CN(C(C3CSCCS3)=O)C2)c[nH]c2cc(F)ccc12 C1(C(N(CC(C)(C)Nc2ccnc(C3CCC3)n2)C)=O)CC(C(C)(C)C)=NO1 CCCC(C)(CC)C(=O)NCCCCN(C(=O)CC(C)N1CCCC1=O)C N1(C(C(C)NC(C)=O)=O)CCOCC(F)(CNC(c2nn(C)cc2[N+](=O)[O-])=O)C1 N1(C(C(CC=C)CC=C)=O)CCC2CN(C(=O)COCC3CCCO3)CCC12 c1(C(=O)NCCCCN(C(=O)CCCCNC(N)=O)C)cccn2nccc12 N1(CCCn2c(C)ncc2)CCC2CCC(C1)N2C(=O)C(C1CCCCC1)=O c1(C(=O)NC2C(C)N(C(=O)Cc3cncc(C#N)c3)CC2)cc(O)cc(O)n1 CC1CCN(C(C23CC(NC(=O)C(O)Cn4cncn4)(C2)C3)=O)CCS1 C1(NC(CCC#C)=O)(CF)CCN(C(=O)C(c2c(C)noc2C)C)C1 C1(C(=O)OC)CC12CCCCC2.C1(CN(CC)CC)CCCN1C(=O)C1CC1 C1(NC(c2ccn(C(F)F)n2)=O)CN(C(c2cnccc2Cl)=O)C2(CCCC2)C1 N1(C(C2CCC(C)CC2)=O)CC2(CNC(=O)CC3CCOC3)CCC1CC2 c1(C(=O)NCC(CC)NC(=O)CC2(C)CCCCC2)c(C)ccn1C N1(C(C23OCC(CC)(C2)C3)=O)CC(NC(=O)Cn2cc(Br)cn2)C2(CCC2)C1 Cc1ccc(CC(N2CC(OCCNC(=O)C(C)(C)C3CCCO3)C2)=O)o1 C1(c2nnnn2C(C)(C)C)(NCc2ccc(SC)cc2)CCC(SC)C1 S(=O)(=O)(c1ccc(F)c(Br)c1)N1C2CN(C(c3cncnc3)=O)CC21 N1(C(C(C)OC2CCOC2)=O)CC2(CC(NC(=O)C3=CCCCCC3)CO2)C1 C1(C)(C(=O)NCCCN(C(=O)C(C(C)C)n2cnnc2)CC)CCCCNC1=O Cc1cc(F)sc1C(=O)NCC(C1CCOC1)NC(c1ccncc1N)=O c1(-c2n(C(CC)C)nc(CS)n2)cccc2ccncc12.O(C(F)(F)F)CC C1(CNC(C2C(C)SCCC2)=O)CCC2(CN(C(c3cnc4n3CCS4)=O)C2)O1 N1(C(C(CSC)C)=O)CCC2CCN(C(C3CCC(C)CC3)=O)CC2C1 C=CC1(C(=O)NC2CCCC(NC(c3csc4nnsc34)=O)CC2)CCCCC1 N1(C(C(c2ccoc2)NC(CCCC2C(C)C2)=O)=O)CC2(C1)CC1(CCC1)C2 Cc1ccc(=O)n(CC(=O)NC2CN(C(C3=C[SH]=CCCC3)=O)CC2CO)n1 CN1CCC(C(=O)NCCc2ocnc2CNC(C2CNC(=O)C2)=O)C1 CCC(CC(=O)NCC1(NC(=O)C(C)(CC)OC)CCC1)C(C)C CN=c1[nH]cc(C(N2CCCC2(C)C(=O)NCC(C)O)=O)s1 C1(N(C(=O)CCc2cn[nH]c2)CC)CCCN(C(=O)C(n2nc(C)cc2C)C)C1 C1(C(N2CC(NC(c3sccc3Cl)=O)C(CC3CC3)C2)=O)CCCC12CCC2 C1(C(=O)OC)CCCCC1NC(=O)COC1CN(C(=O)C(F)OC(F)(F)F)C1 N1(C(CN(CCOC)C)=O)CC(C(=O)NC(CC)CC(=O)OC)CC12CCC2 c1(C(=O)NCC23C(CN(C(C4(COC)CCCO4)=O)C2)C3)occ2c1CCOC2 c1(COC)cc[nH]c1C(=O)NC(C)(C)C(=O)Nc1cccnc1 c1(C(N2CC(NC(CNS(C)(=O)=O)=O)NCC2)=O)ccc2c(Br)nn(C)c2c1 C(=O)(C1=NN2CCCN=C2N1)NCC(C)NC(c1cnc(CO)s1)=O CCCCC(O)CC(=O)NCCCCC1CN(C(=O)CCc2cnn(C)c2C)C1 Cc1cc2[nH]c(C(=O)NC(C)CN(C)C(C3CCCC(O)C3)=O)cc2o1 c1(C(N(C2CC3CN(C(C(CC=CC)C)=O)C2C3)C)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C1(C(=O)NCCc2ccc(C)cc2)CC2CN(C(=O)CCC3CC3(C)C)CC2C1 C(C(C(=O)N1CC(CNC(=O)CSc2nnnn2C)(OC)C1)OC)OC c1(C(N2C(CNC(CC3CC(=O)NCC3)=O)CC(F)C2)=O)cccn2cnnc12 c1(C(N(C2CCN(C(C3CC34CC4)=O)CC2)CC#C)=O)cc2ncn(C)c2cn1 CC1CC2(CCN(C(C3CCCC(C#N)C3)=O)CC2)CN1C(c1cc(Cl)no1)=O Cc1nn(C)c(C(N2CCCCC(NC(c3cccc(N)c3C(F)F)=O)C2)=O)c1Cl c1(C(=O)NCC2CC(O)(CNC(C3(O)CCC3)=O)C2)cc(Cl)ccc1O C(=O)(CCC1=NNC(=O)CC1)NC1CC(CNC(C2(C)C(C)C2)=O)C1 C(=O)(CC(C(F)(F)F)NC(c1ncc(F)cc1N)=O)NCCc1nc(CC)on1 N1(C(C2CCC(=O)N2)=O)CCCC(NCc2ncsc2Br)C1 C=CCCC(C(=O)NC1CCCC1)NC(=O)CO.C1(O)(CCN)CCC1 CCCCC(CC)C(=O)NCCCNC(c1ccc(NC(=O)OC)cn1)=O C1(O)(C(=O)NCC(C)NC(c2cccc(C(N)=O)n2)=O)CCOC1(C)C N1(C(Cc2cnc(C)nc2O)=O)CCCC2(NC(=O)Cc3cccs3)CCCC12 C(=O)(C(C)C(C)NC(c1sncc1C)=O)NCC=CCCOC N1(C(C=CCOC)=O)CCCC(C)(NC(c2c(C(F)F)cccc2C(F)F)=O)C1 c1(C(N(C2C3CN(C(=O)CCNS(C)(=O)=O)CC23)C)=O)nccnc1Cl c1(CNC(C(CN(CC)CC)F)=O)cccc(C(=O)NC2CC(C(N)=O)C2)c1N C1(C(N(C)CC2(O)CCN(C(C3(COC)CCC3)=O)C2)=O)CC2CCC(C1)O2 n1(CC(N2C(C)CC(CNC(C3(CO)CC3)=O)C2)=O)ncc2cccnc12 Cc1nn(CCO)c(C)c1C(N1CC2(NC(c3cncc(F)c3)=O)CC1C2)=O c1(OC)ccc(NC(C2CCCN(S(=O)(=O)CC(C)C)C2)=O)cc1Br C1(C)(C(N2CC(NC(N(CC(c3ccccc3)O)C)=O)C2)=O)CC1(F)F c1(CN(CC)CC)ccc(C(=O)NC2C(NC(C3(CC)CC3)=O)CCC2)cc1 C1(CNC(C=C(C)Cl)=O)CCC2(CN(C(=O)CCOc3ccccc3C)C2)O1 Nc1ccc(C(N2CCCCC(CNC(C3CC3(Cl)Cl)=O)C2)=O)nc1F C(N=c1[nH]c(N2CCCOC(C3CCC3)C2)nc(=N)[nH]1)C1(F)CC(OCC)C1 N1(C(C2N(C)C(=O)NC2)=O)CCCC2(C1)CN(C(=O)C(c1cncn1C)O)C2 Cc1ccc(SCCN(CC(F)(F)F)C(=O)NC(=O)C=CCF)o1 CCCCCCCn1cc(CC2CCN(C(C3CC(C(F)(F)F)C3)=O)C2)nn1 C12(C(=O)NCC3CCC(C)CO3)CC(CN(C(=O)C(C)CC#N)C1)C2 C=CC1CCCC(C(=O)OC(C)(C)C)C1.C12CCN(C1)C(=O)CONC(=O)CO2 c1(CNCC23OC(C)C(C2)C3)c(F)ccc(F)c1Br c1(C(=O)NCC)ncc(C(=O)OC(c2cn[nH]c2)C2COC2)o1 C1(COC)(NC(=O)CC2CCOCC2)CCCN(C(=O)CC2CSCCO2)C1 Cc1cc(NC(C2(NC(=O)C(C)CO)CCC(C)(C)C2)=O)cc(O)c1 C(C(C)(C)C(=O)NCC1CC(NC(C2CC3(C2)CC3F)=O)C1)SC N1(C(c2ccc(NC)cn2)=O)CCCC(NC(c2cn(C(C)C)cn2)=O)CC1 N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C(c2cc(C3CC3)n(C)n2)=O)CC1C N1(C(c2c(C)nn(CCC)c2C)=O)CCCC2C1CCN2C(C1CC1CF)=O C12(CC(=O)NC(CCOC)CNC(=O)Cc3c[nH]nc3O)COC(CF)(C1)C2 c1(C(=O)NOC2CCC2)ncoc1CNC(c1ccc(CO)o1)=O O=C(CC1CCN(C(c2sccc2CO)=O)CC1)NNC(=O)NCc1ccccc1 c1(-c2cn(CC(F)CO)nn2)ccc(F)cc1.c1(C(C)C=O)ccc(Br)cc1 C(=O)(CCC(C)(F)F)NCC12OCC(NC(c3ccc(CC)[nH]3)=O)(C1)C2 CC1CN(C(c2cccc(CS(N)(=O)=O)c2)=O)CC(C)N(C(=O)CNC(N)=O)C1 N1(C(c2ccc(OC)o2)=O)CCCC2(CCCCC2NC(c2oncc2C)=O)C1 c1(C2(C(=O)NCC3CN(C(C4CCC(C)O4)=O)C3)CCC2)ccccc1Cl C1(NC(C2(CC)CCOCC2)=O)CCC2CC1CN2C(C1CCC(CC)CC1)=O C(=O)(C(F)(F)CCn1ccnn1)NCC1(CNc2cc(COC)ncn2)CCC1 C(=O)(C(O)CC(C)(C)C)NCC(CNC(c1cnc(C(C)O)s1)=O)(C)F N1(C(C2C(C(=O)Nc3c(C)cc(F)cc3)C2)=O)CCC2C(C1)NC(=O)N2C c1(CC(=O)NC2CC23CC(NC(C2(O)CC2)=O)C3)c[nH]ccc1=O c1(C(C(=O)NCCSC)N(C)CC2CCOC2(C)C)sc(Br)cc1C C12(CNC(C(C3CCN(C(CSCCC)=O)C3)C)=O)COC(COC)(C1)C2 CC(C)(CNC(=O)CCOC(C)(C)C)CNC(C1CN(C(C23CC(C2)C3)=O)C1)=O C1(C(=O)NC2CCCC(NC(C3CN(CC)C(=O)C3)=O)C2)OCCN(C)C1=O C1(NC(C2CC(O)(CC#C)C2)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1F C1(C(=O)NCCC2CC(NC(c3nnn(C(C)(C)C)n3)=O)C2)(CC)CCOC1 N1(C(=O)C(O)CC2CC(F)(F)C2)CC2CC1CN2CC1(c2cccc(F)c2)CC1 C(CCCCCC(=O)N1CCC(O)(CN(C(=O)CN2CCC(C)(C)C2)C)C1)SC N1(C(C(CCOC)(C)C)=O)CCN(C(C23CCC(CC2)C3(C)C)=O)CC(O)C1 c1(C(C)C(=O)NCc2nc(-c3ccco3)n[nH]2)ccc(F)cc1F Cc1cc(C(=O)NCCNC(=O)NC2C3CCC2(c2cncs2)C3)cc(N)c1 C(N=c1ccnc(N2CCOCC(C)C2)[nH]1)C1N(CC)CCC1 C1(NC(C2(CNC(C3CCCCC3F)=O)CCC2)=O)CCCN2CCCC12 Cc1cc(C(=O)NCC2(C)CCCN2C(C2CC(F)(F)CS2)=O)cn(C)c1=O C(C(COC)CC(=O)N(CCC(C)NC(=O)CCC(C)(F)F)C)OC C1(NC(C2C(C(=O)NCC#C)C2)=O)CCN(C(=O)CC2=CCCC2)CC12CCC2 C1(CNC(CC2(C)CCCO2)=O)CCN(C(=O)CCCC2(O)CCOCC2)CC1 CC1(C)CN(C(C2CCOCC23CCC3)=O)CC(CNC(=O)CN2CC=CC2)O1 c1(C(N(CC(NOC(CC)C)=O)CC2CC2)=O)cc(C)c(C)nn1 S(=O)(=O)(c1ccc(C)cc1)NCCC(=O)NC(CN(C(C(CCC)OC)=O)C)C C1(NC(N(C2CN(C(C(C)Cc3ccco3)=O)C2)C)=O)CCCCCC1 N1(C(C(C)CS(C)(=O)=O)=O)CCCC(N=c2nnn(C)[nH]2)CC1 C12(NC(N(C)CCN3CCC(c4cc(F)ccc4F)C3)=O)CCCCC1OCC2 C(C(C(=O)N(C)CC1CC1(C)C)N(C)C)NC(C(C1CCC1)OC)=O C1(CC)CN(C(=O)C2=C(Cl)CC2)CCC1NC(=O)Cc1cnsc1 C(=O)(N=c1[nH][nH]c2c1CN(Cc1ccc(Cl)c(I)c1)C2)c1ccc(C)c(F)c1 C(=O)(CCCC(F)(F)F)NCCC(C)(C)C(=O)Nc1cccc(OCF)c1 O=S(=O)(c1cccnc1NC)NC1CC1C1CC1.N1(CCN)CCSCC1 N1(Cc2c(C)c(F)ccc2)CCC2(CCN(C(C3CC34CC4)=O)C2)C1 C(CCCCC(=O)NC1CCN(C(c2cccc(C#N)n2)=O)CC1F)N(C)C N=c1[nH]c(C2CC2)ncc1C(=O)NC1CCC1NC(C1CCNC1=O)=O N1(C(CCC=CCC=C)=O)CCCCC(CNC(=O)Cc2cc(Cl)sc2Cl)C1 CCC(C)CCCCC(=O)N1CC(OCC(N2CCC23CCSCC3)=O)C1 N1(C(C23N(C(c4c(N)cncc4)=O)CCC2C3)=O)CC2(CCC1CO)CC2 N1(C(C2CCCCC2(F)F)=O)CC2CCC(C1)N2C(C1CCc2c[nH]nc2C1)=O C=C(C)CC(C(=O)Nc1ccc(C(=O)NC2CCCC2)cc1CC)OC C12(CNC(=O)CCF)CN(C(c3cn(-c4ncccn4)cn3)=O)CC1CCO2 CC1C(NC(c2ccnc(-c3ccccn3)n2)=O)CCN1C(C1CC(F)(F)C1)=O C(C(C)(C(=O)NOCC1CCC1)NC(C1CCN(C)CC1)=O)SC CC(C)CC(C(=O)N1CCOC2CC12)NC(=O)CCNC(=O)CO C(=O)(CC(C)(C)C(=O)NC1(CN(C)C(C2CC(OC)C2)=O)CC1)OC C1(C(C)O)CN(CCC2(c3cccc(Br)c3)CC2)CCO1 Cn1ccc(C(F)F)n1.C(=O)(CC1CC1CN(C(=O)OC(C)(C)C)CC)O CCC(CNC(c1ccc(S(C)=O)cc1)=O)N=c1[nH]c2c(C)cccc2o1 O=C1CC(=O)CC(C(=O)NC2(C(=O)NC3CCN4CCCCC34)CC2)C1 c1(NC(C)=O)ccc(F)c(C(=O)NC2CCCCC2CNC(=O)CC(C)F)c1 CCCCCC(O)C(=O)NC12CC(C(N3CCS(=O)C(C)C3)=O)(C1)C2 CC1CC(=O)CCC1C(=O)N(CC(C)(C)CNC(C12CC3CC1C2C3)=O)C Fc1ccccc1CNC(=NCC1CC1(Cl)Cl)NC1CCOCC1 c1(C(=O)NCCCCCCNC(C(C)CO)=O)c[nH]c2cccnc12 N1(C(CC2CC(NC)C2)=O)CC(C(=O)Nc2cccc(OCF)c2)C(C(C)C)C1 O(NC(=O)C(C1(O)CCCCC1)NC(c1ccc(Cl)cc1)=O)Cc1cn(C)nc1 C(N=c1[nH]c(N2CCC(C(N)=O)C2)nc(=N)[nH]1)c1ccc(NCC(C)C)cc1 N1(C(C#CC(CNC(CC=C(C)C)=O)(C)C)=O)CCC2(CC1)CN(C)C2 C1(CNC(C2CCCN(CC)C2)=O)CN(C)CCN1C(C1OCCO1)=O C1(C(=O)NC2CCN(C(=O)C=C(Cl)Cl)CC2CO)Cc2ccccc2CO1 N1(C(c2c(C)scn2)=O)CC2CC(C(=O)NCC(C)(C)C(C)C)CC2C1 Cc1cc(CNC(=O)Nc2cccc(C(=O)NC3(c4ccco4)CC3)c2)ccn1 CC1(C(N2CCC(C(CO)NC(=O)C=CC3CC3)CC2)=O)CC2CC2C1 C1(OCC)CC2(C1)CC2.C(=O)(CCCN1CCCC1)NC(C)CN(C)CCOC C(=O)(CN=S(C)(C)=O)NCC1CC(OC)CN1C(C1CC(=O)N(C(C)C)C1)=O N1(C(C=CC(CC)C)=O)CCC(CN(C(=O)CN2CCCNC2=O)C)CC1 N1(C(C(C(C)C)F)=O)CCCN(C(=O)CC2CC2)CC1C C(C(C)(C)C(=O)NC1CC(O)(C(=O)Nc2ccc(N3CCNC3=O)cc2)C1)OC C1(NC(CC(OCC)OCC)=O)CCCCCN(C(=O)C2=CCCCC2)C1 Cc1[nH]ccc1C(=O)NC(C(=O)NCC(c1ccccc1)C)C1CCCO1 C1(C(=O)Nc2c(C)csc2)CN(C(=O)CCc2cn[nH]c2)CC1C CCCCC(O)C(=O)NC(C)(C)CNC(c1cc(C(F)F)cs1)=O N1(C(c2c(NC)cccc2)=O)CCC2CC(C1)CN(C(=O)Cc1scnc1C)C2 c1(NC(C23C(CN(C(C#C)=O)C2)C3)=O)cn2ncccc2n1 C(=O)(CC1=NNC(=O)C1)NC(CC)CNC(c1nccc(Cl)c1F)=O c1(C(N2CC(F)(C(=O)NC(CCC)C(N)=O)C2)=O)c(C)oc(C)c1C C(=O)(CC(C)CC(F)(F)F)NCCOCCNC(C(C1CCC1)OCC)=O N1(C(CCC2CC(C)C2)=O)C(CNC(c2csc(Cl)n2)=O)CC2CC12 c1(CNC2C(C)CN(C(=O)OC(C)(C)C)C2)oc2ccccc2c1CO C(C1CN(C(=O)Cc2ccnc(O)c2)CC1C(=O)NCCCOCCCC)=CC Cc1ccc(C(N2CC3CCC3(C(N3CCC(F)C(F)C3)=O)C2)=O)c(C(F)(F)F)c1 N(C(=NCC(C)N1CCOCC1)NCc1cccc(Cl)c1)Cc1c(C)ccs1 Cc1ccc(NC(=O)C(C)(C)NC(C2CC2(C)C)=O)c(O)n1 Cc1nn(C)c(C)c1CC(N1CCC(NC(c2cccc(=O)o2)=O)C(O)C1)=O C1(C(=O)NCC2(F)CC(CNC(c3ccc(O)nc3)=O)C2)COC2(CCC2)C1 Cc1ncc(CCC(=O)N(C)CCN(C(=O)C(O)C2CCCC2)C)s1 C12(CNC(c3cnc(S)[nH]3)=O)CCCC1CCN2C(c1coc(C(F)(F)F)c1)=O N1(C(c2c(C(C)C)scn2)=O)CC(CNC(C2CCC(=O)NC2)=O)C(C)(C)C1 C1(OCC)=CC=C(NNC(=O)N=c2[nH]nc3ncccc3n2)C1 CC1(C)CN(C(C2CC2C2CCC2)=O)CC1CNC(c1cnc(S)n1C1CC1)=O c1(C(N(C2CCN(C(C3CC(F)C3)=O)CC2)CC)=O)ccc2nc(O)oc2c1 c1(C(N(C2CCN(C(=O)C(C3CC(F)(F)C3)O)C2)CC)=O)ccn2c1CSCC2 c1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)ncn2c1CCC2 C1(N(C(CNC(CCC)=O)=O)C)CCCCN(C(=O)C(C)=C(C)C)C1 N(C(=NCCCC1CCC1)NCC1CCCO1)CC(c1c(C)nn(C)c1C)O CC(CC(=O)NCC1CC(C)CCN1C(C1CC(N(C)C)C1)=O)C(C)(C)C N1(C(C(CC)n2cccn2)=O)CCC(C(CO)NC(=O)CN(C)CC)CC1 C1(CC=C)(NC(=O)C(C)CC)CCCN(C(=O)CC(=O)OCC(C=C)O)C1 CC1=C(C(=O)NC2CCCC(NC(=O)CC(C)CNC(=O)OC(C)(C)C)C2)CCC1 c1(NCc2cn(C)nc2)cc(-c2ccnn2C2CCC2)ccn1 c1(C(=O)NC(C2CCN(C(C3CC(OC)C3)=O)C2)C)ccc2ncn(C)c2n1 CC(C)(CNC(c1cnc(S)nc1)=O)CC(=O)NCC1(O)CC1 Cc1cccc(C2CCCN2C(=O)C(=O)N(C)CC2CCN(C)CC2)c1 C(C(C)(C)CC(C)C)c1nc(CC)on1.N12CCCC1C=CCOCC2=O C1(=O)C(C(=O)OC)N1C(C)C(=O)N(C(C)CC(N)=O)C.CCCOC CCC(CC(F)F)C(=O)NCCCCN(CCCNC(=O)CCC1CC1(F)F)C c1(C(N2C(c3scc(C)c3)CCC2)C(=O)NC2CC2)nc(C)c(C)n1C C(=O)(C(=O)N=c1cc(C)o[nH]1)N1C(C)CC2CN(C(C(C)SCCCC)=O)CC21 CN1CC2CCN(C(C34CCC(NC(=O)CCCC#N)(CC3)C4)=O)C2C1 Cc1ccncc1C(N1CCC(OCCNC(=O)C(O)C2CC2)C1)=O C1(NC(c2cnc[nH]2)=O)C=CCN(C(C2(C(F)(F)F)CCOCC2)=O)C1 CCCC(CCC)=CC(=O)NCCCN(C1CCCC1)C(=O)CC1CC(F)(F)C1 c1(CCC)cc(C(=O)NC(C)(C)CCCNC(c2cnsc2C)=O)c(C)o1 C(=O)(C(CCCC)N(C)C)NCC(CCCC)NC(=O)CCCCN(C)C(C)C CCC(CCC(=O)N(C)CCc1cnc[nH]1)NC(=O)CSC1CC1 C1(N(c2cnc(F)nc2)CC)COC2C(C(=O)OCC)COC12 c1(-c2n(CC=C)nc(Cc3cccnc3)n2)ccnc(OC)c1Br C1(C(C)C)CN(C(c2sc(-c3ccccc3)cc2Br)=O)CC(=O)N1 N1(C(Cn2c(C)cc(O)cc2=O)=O)CC2(C)CN(C(=O)C=CCF)CC2(C)C1 C1(CCNC(c2ccc(C(CC)C)cc2)=O)CC(F)(F)CN1C(=O)CCCSC C(=O)(C(C)C(O)C(C)C)NC(CC)CC(=O)NCC1C(C)C1C c1(CC(N2CCOCC2CNC(C2(F)CC=CC2)=O)=O)ccc(OC(F)F)cc1 N1(C(CC(C)OC)=O)CCOc2ccccc2C1CO Cc1ccc2n[nH]cc2c1C(=O)NCC1CCN(C(=O)CC(C)O)CC1(F)F C=CC1(C(N2CCCC2CC(N)=O)=O)CCN(C(=O)C(C)(C)C(=O)OC)CC1 C(c1c(F)cccc1F)=CC(=O)NC1CC1NC(=O)C(O)Cn1cncn1 c1(C(C)NC(c2c(CNC(CSCC(=O)OC)=O)n[nH]c2)=O)ccc(C)cc1 c1(C(=O)NCCC2CC(NC(c3cnc(C(=O)OCC)s3)=O)C2)ccnc(O)c1 C1(C(=O)NC2CN(C(CC)=O)C2)CC2CC1CC2NC(c1cn(C)ccc1=O)=O C1(C2CN(C(c3ccnc(-n4cncn4)c3)=O)C2)(NC(c2c(C)[nH]cc2)=O)CC1 C1(=O)CC(C)OCCN1C.C(=O)(CN(C(=O)C=CCOC)C)OC CCC(N=c1nc2c(ncn2CC)c(NCCC(F)(F)F)[nH]1)C1CCC1 N1(C(c2ccc(C)cc2)=O)CCC(NC(c2cncc(N)c2C)=O)C2(CCC2)C1 C1(C(N)=O)CCC2(CCC2)C1NC(=O)CC1CSC1 C(C(C)C)(C(O)C(=O)N(C1CC(NC(=O)C(C)Oc2cccnc2)C1)C)OC Cc1cnc(C(N2CCC(C3CCCN3C(=O)C(F)C3CCC3)CC2)=O)cn1 CCCC(C)(C)CC(=O)NCCC(C(C)C)NC(c1cc(N)c(OC)cc1F)=O N1(C(C2C(CCC)C2)=O)CCCC2(CCCN2C(c2csc(C)c2C)=O)C1 N1(C(C=CC(=O)OC(C)(C)C)=O)CCC(NC(c2ccc(CO)cc2)=O)C12CC2 Cc1ccc(C)n1CCC(=O)NCCSCc1cn(-c2ccncc2)nn1 C(=O)(CC(C)C(C)(C)C)N1CC(CC=C)(NC(C23CC(C)C2C3)=O)C1 c1(CC(C)NCC(c2cc(O)ncn2)O)cccc(Cl)c1 Cc1cccc(Cl)c1C(c1nnnn1CC1CC1)NCCC1CCS1 N1(C(C2CCC(C(N)=O)O2)=O)CC2(CCC2NC(=O)C=Cc2cocn2)C1 C1(C)(C(N2CCCC(C3N(C(CCC(C)C)=O)CCCC3)C2)=O)CCOC(C)C1 c1(NC(C)=O)cccc(C(=O)NC(C2CCCN2C(c2csnn2)=O)C)n1 Cc1nc(CO)sc1C(=O)NCC(C1CCN(C(C2(C)COC(=O)N2)=O)CC1)F c1(C(=O)NC(CNC(CNC(CC)=O)=O)CO)nc2ccccc2nc1C C1(NC(C(n2ccc(C)n2)C)=O)CN(C(=O)C(F)(F)C2CC2)CC(F)(F)C1 O=C(Cc1cccs1)C(=O)N1CC(CNC(C2CCC2c2nc[nH]n2)=O)C1 c1(C(=O)NCCCCNC(C2(F)C(C)C2)=O)sc(Br)cc1Cl c1(C(=O)NC(CN(C(=O)CC2CC2(Cl)Cl)CC)C)ncc(C(N)=O)cc1Cl c1(CNC(C2N(C)c3ccc(Br)cc3NC2)=O)ccc2cc(S(N)(=O)=O)ccc2c1 C1(C(=O)NCC(C)NC(c2c(Cl)ccc(C)c2)=O)Cc2ccc(Cl)cc2C(=O)O1 c1(C(N2CCC3(NC(=O)Cn4ncnn4)C(C2)C3)=O)cc(Cl)cc2cccnc12 C1(C(=O)NC(C2(O)CN(C(C(CCCC)O)=O)C2)C)CN2CCN1C(C)C2 CCCCCNC(C1(CNC(C2CC(F)C2)=O)CCC1)=O c1(COC(C)C(=O)Nc2ccc(F)c(Br)c2)ccc(=O)n(CCO)c1 C1(NC(C=C(CC)C)=O)CN(C(c2cnn(C)n2)=O)C(C)(CC)C1 N1(C(c2cccc(N)c2)=O)CC2CCC(NC(c3ccc(C(N)=O)s3)=O)CC2C1 C(C(C)(C)C(=O)N1CC(C)(NC(=O)Cc2nc(C)sc2C)C1)SC C(=O)(CCS(C)(=O)=O)NC(CNC(CCNC(=O)OCC)=O)CC n1(CC)nc(C(=O)NCC2CC(CNC(=O)C(C)(CC)OC)C2)cc1O Cc1ccc(CNC(N2CCC(=Cc3cccc(F)c3)CC2)=O)cc1C#N c1(CC(=O)O)ccc(CN(C(=O)CC2CC2)CCN(C)C)cc1 c1(-c2cn(CCC(N3CC(CCCC)OCC3)=O)nn2)ccnc(F)c1C c1(C(N2CC(N(C(=O)CC3CCCCO3)C)C3(C2)CC3)=O)ccc(Cl)c(F)c1N CC(CC(C)(C)C)N=c1[nH]c(=NCc2nn[nH]c2C(C)(C)C)[nH]c2c1COC2 c1(CC)noc(C(C)NC2CCCC2Cc2cncn2C)n1 CC(CCCCNC(=O)C(C)(O)C1CCC1)NC(=O)C(C)(C)CO N1(CC)C23CCCC2CC1C3.N1(C(=O)OCC)CCN(C2CN(C(=O)O)C2)CC1C C(CCCC(=O)NCC1CC(NC(=O)C(F)CC2CC2)CCO1)N(C)C c1(OC)ccc(C(N2CCC(NC(=O)CC3CCCN3)CC2)=O)cc1N n1(CC)c(C)cc(C(=O)OC(C)C(=O)Oc2ccc(C(=O)NC(C)(C)C)cc2)c1C C1(CNC(CCSCCCC)=O)CC2CCCC2N1C(=O)Cc1nc[nH]n1 CN1C(=O)CCC1C(=O)NC1CC1NC(c1ccc(N2CCNS2(=O)=O)cc1)=O Cc1c(C(C2(C(N3CCCC3CNC(=O)CC=C(Cl)Cl)=O)CC2)=O)cccc1F CC(C)(CNC(C1(C)CCCN(C(=O)CCN2CCCC2)C1)=O)CCCO N1(C(c2c(OC)nc(C)cn2)=O)CC2CCC1CN2C(=O)CO C(CC(CC)C(=O)NCC12CC(CO1)N(C(C1(SC)CCC1)=O)C2)=CC c12[nH]ccc1CNC2=O.C1(NC(C2CC(OCC)C2)=O)CCN(C)C1.COC c1(C(=O)OC)coc2cc(C(=O)NCC3(O)CN(C(=O)C(C)C(C)O)C3)[nH]c12 c1(CNC(c2cccc(OC(C)C)c2)C)c(OC)cccc1O c1(NC(N2CC(C(Cn3cc(CC(C(C)C)O)nn3)F)C2)=O)ccc(Cl)c(Cl)c1 Cc1nscc1C(=O)NCC1OCCC1C(=O)NOCC(C)(C)C c1(C(=O)NCC2N(C(c3c[nH]c(=N)o3)=O)CC=C2)n[nH]c2ccccc12 c1(-n2cc(C(=O)NCc3onc(CC(=O)O)n3)nn2)ccccc1Cl c1(OC)cc(C(=O)NC(C)(CNC(c2nnc(S)n2C)=O)CO)cc(F)c1F N1(C(CN(C(=O)OC)C)=O)CCN(CC(C)NC(C2CCC(=O)N2)=O)CC1 c1(C(=O)NC2C(CNC(c3nc(COC)[nH]n3)=O)CCC2)cc(C)cnc1C N1(C(CC2CCN(C(CCC=C)C)C2)=O)CC2CC1C1OCCOC21 c1(CC)sc(C(=O)NC2CN(C(=O)COc3cn[nH]c3)C2)cc1C C1(CC(=O)NC2COCC2CNC(c2cc(Cl)cc(Cl)c2)=O)CCC(F)(F)CO1 CC1CC(F)CN1C(=O)Cn1cc(C2CCC2)nn1 N1(C(C(C(C)OC)NC=O)=O)CC2CCC(C1)N2C N1(CC(=O)OC(C)(C)C)CSCC1=O.C12CC(C1)CC(=O)N2C(=O)C=C(C)C(F)F C(=O)(CC(C)(C)C(C)=O)N1CCC(N(C(CCCC#C)=O)C)C(C)C1 N1(C(Cc2c(C)non2)=O)CCOCC1CNC(c1ccc(Cl)[nH]1)=O C(CC(=O)NCC1(F)CCN(C)C1)(C(F)F)NC(c1c(CC)occ1C)=O C#CCC(C)(C)C(=O)N1CCC2C(C(=O)NC(C)(C=C)CC)C2C1 c1(NC(=O)CC2CCCC2)cnc(CN)nc1.N12CCCC1CN(C)C(C)C2=O N1(C(C2(CCOC)CCC2)=O)CCC(NC(c2cn3c(n2)CCC3)=O)C(CO)C1 N1(C(CCN(C)C(C2CCCOCC2)=O)=O)CC(O)CC1C(N)=O C1(C(=O)NCCC2CN(C(CCC(=O)OC)=O)C2)CC2CC(O)CC(C1)C2.C(=O)OC c1(COC(c2cnc(C3CC3)nc2)=O)noc2ccc(Br)cc12 c1(C(N2CC(C)C(NC(=O)C(CO)c3ccccc3)C2)=O)cc(Br)ncc1Br Cc1ccc(C(=O)NC(C)C(C(C)C)NC(c2cnc(O)n2C)=O)nc1O C1(NC(C=NOC)=O)C=CCN(C(C2CC23CC3)=O)C1 c1(C(=O)NCC(C)(O)CNC(C2(Cl)CC2(F)F)=O)nccc2c1CNC2=O N#Cc1nc(NC(=O)C(N2CCC(C3CCCO3)CC2)=O)cc(Cl)n1 S(=O)(=O)(c1ccc(=NCc2ccco2)[nH]c1)N(CCCOC)C N1(C(C(C)SC)=O)CCC2C(NC(=O)CCN3CCOCC3)C12 c1(CC(=O)NCC2(F)CC(CNC(CCC(=C)C)=O)C2)c[nH]c2c(C)cccc12 N1(C(CC(C=C)C)=O)CCC2CN(C(c3csc(C(C)(C)C)n3)=O)CC2C1 N1(C(CN(C2CCCC2)CC(C)C)=O)CCC(NC(=O)Cn2cnnn2)C12CC2 c1(C(=O)OC(C2CCOC2)Cc2ccccc2)cc(C2CC2)n[nH]1 c1(C(N2CCOCC(NC(C(F)OC)=O)C2)=O)cc2n(n1)CC(C)(C)CO2 Cc1ccc(O)c(C(=O)NCCC(C)NC(=O)C(C)Cc2ccnn2C)c1 c1(N(C)CC2(OC)CCOC2)nc(NCC2CCC3(CC3)C2)c2c(ncn2C)n1 c1(CC)c[nH]nc(C(=O)N(C(C)(C(=O)NC(C)C)C2CC2)C)c1=O c1(C(=O)NCCC(C)NC(=O)C(C)(C)Oc2ccc(F)cc2)ccc(C#N)o1 N1(C(C2N(C)CSC2)=O)CCC(F)(CNC(C2CC23CC3)=O)CC1 Cc1c(C(=O)NC(CNC(C23CCC(CC2)C3)=O)C2CC2)c(C(F)(F)F)nn1C N1(C(C2N(CCC)C(=O)CC2)=O)CCC2CN(C(=O)CC(C)(C)O)C2C1 C(=O)(C1=CCCCCC1)N1CCN(C(C(C)CC2CC2)=O)CC1CC1CC1 C(=O)(C1=CCC(C)CC1)NCC.N12CCOCC1C(=O)N1CCN(CC1)CC2 C1(C(C)NC(C(C)Cn2ccnc2)=O)CCN(C(C2(c3nccs3)CC2)=O)CC1 N1(CC2C(C(=O)NC3CCCC3)CC2)CCC(NC(COCC(=O)OC)=O)C1 C1(COC(=O)CCSCC(=O)Nc2ccccc2)C2CC3C(C2)C13.c1cccs1 c1(C(=O)NCC(CCCC)NC(=O)C(C)OCCOCC)ccc2nnnn2c1 CC(CCNC(C1(NC(=O)CCCOC(C)(C)C)CCCC1C)=O)C(F)F N1(C(CCC(=O)NCC)=O)CCCC(O)(CNC(C2CC2C(C)(F)F)=O)CC1 C1(NC(Cc2cn(CC)nn2)=O)CN(C(=O)C(O)CC2CCCC2)CC1C c1(C(N(CCC(C)NC(=O)C2CC2)C)=O)cccc(O)n1 C(=O)(C(C)(C)CC1CCOCC1)NCC(C1CC1)NC(C=CC(CC)C)=O N1(C(C2CC(C)(C)C2)=O)CCC2(CCCN(C(=O)COC(F)(F)C(F)(F)F)C2)C1 C1(NC(C(CC(C)C)(C)O)=O)CN(C(=O)C=CC=C(Cl)Cl)CC12CCOCC2 C1(C(=O)NC2(CNC(C3C(C(=O)OC)C3)=O)CC2)CC1(C)C N1(C(c2c(CCC)nns2)=O)CCC2CN(C(=O)C(C)P(C)(C)=O)CC2C1 c1(NC(c2cnn3c2OCC3)c2n(CC=C)nnn2)cc(C)cnc1C CC1(C(N2CC(CC3(NC(c4cocn4)=O)CC3)C2)=O)CC1Br C1(NC(c2cc(C)ncc2)=O)CN(C(c2nn(C)c(C)c2Br)=O)CCC1F N1(C(CC2C(CNC(=O)CCn3ccnc3)C2)=O)CCC(CN2CCC2)C1 C1(CC)CN(C(=O)CSC(F)F)CCN1C(c1cccn1Cc1ccccc1)=O c1(C(=O)NCCN(C(C(CO)OC)=O)C2CC2)coc2c1COC2 CCC(C)C(O)C(C)C(=O)N(CC(C)C(=O)NCCC(C)C)C C1(C(N(CCC(C)O)C)=O)CCCN(C(c2ccncc2)=O)C1 C1(C(C)C)CC(CNC=O)CN(N2CCCC2C(F)(F)F)C1 c1(NC(C2CCS(=O)(=O)N2)=O)nnn2c1COCC2 CC(C(C)(C)O)N(C(=O)C=CC(C)NC(=O)CCC1CCCN1C)C C1(C(c2nnnn2Cc2cccs2)OC)(NCC(c2ccncc2)C)CCSC1 N12CCC(C(c3cn[nH]c3)C1)CNC2.C1(CC)(CC(N)=O)CCCCC1 c1(C(N2CC(F)(C(=O)NCC3(C)CNC(=O)O3)C2)=O)cccc(C#N)c1 C(C)(CCN)OC.C1(=O)CCNCC2(CC2)C(=O)N(C)CCOCCN1C.C(C)(=O)O CC1CN(C(=O)CCSCC(N)=O)CCC1CNC(=O)CCC1CCCN(C)C1 c1(C(=O)NCC2(O)CN(C(C3CC(C)NC(=O)C3)=O)C2)cnn2c1CC(C)CC2 C1(CC(=O)NCC(O)CCNC(=O)CN2CC=CC2)CCC12CCC2 C(=O)(CCC(C)CN(C)C)NC(C(=O)NC(C)C(C)(C)CO)C1CCC1 N1(C(=O)C(C(C)(C)C)=O)CCc2onc(CCC3N(CSCO)CCCNC3=O)c2C1.O c1(C(=O)NC(CCN(C(CCCCSC)=O)C)C)cc(C)c(C)cc1Cl C(CC(=O)N1CCCC1CN(C(=O)C(C)S(C)(=O)=O)C)(C1=CCCC1)OCC c1(OC)ccc(CCC#N)cc1C(=O)N(CCNC(c1cccc(C)c1)=O)C1CC1 C(C)(N=c1nc[nH]s1)C1CCCN(C(C=CCN(C)CC)=O)C1 C1(C(=O)NC2C(NC(CCNC(=O)NC)=O)CC2)CCc2nc(C)ncc2C1 c1(NC(C2(CNC(C(CC=C)CC)=O)CCCO2)=O)cncc([N+](=O)[O-])c1 Cc1nc(C2CC2)oc1C(=O)NCC(C)(F)CNC(=O)CC(C)(C)C N1(C(C(C2CCCO2)NC(c2ccncc2)=O)=O)CCOC(CC2CC2)C1 C1(NC(CNS(CC)(=O)=O)=O)CN(C(=O)C(F)n2ccnc2)CC12CC2 N1(C(c2c(C)nc(CO)o2)=O)CCN(C(=O)COCCOC(C)C)C(C(F)F)C1 CC(CC1CCCC1)C(=O)N1CCCC1CN(c1ncns1)C c1(C(=O)NCC2C3CN(C(C(=O)NCC)=O)CC32)cccc(OC(F)(F)F)c1F c1(C(=O)NC(CNC(C=CC(CC)(C)C)=O)C2CCC2)ccc(Cl)c(Cl)c1O C1(N(C(C(=Cc2ccccn2)C)=O)C)CN(C(=O)Cc2nonc2C)CC1(C)C Cc1cccc2c(C(=O)N(C)Cc3cn(-c4ccccc4Cl)nn3)cnn12 c1(C(=O)NC2CCC(CNC(=O)CSC(F)F)C2)cc(F)c(F)cc1I c1(COCC)nc(Cl)cc(=NC2CCN(C(=O)C(O)C(C)CC)CC2C2CCO2)[nH]1 c1(OC(C)C)ccnc(CNCC#CC2CC2)c1 c1(C(N(C(C)CNC(c2cc(Br)co2)=O)C)=O)ncccc1O Cc1cc(C(=O)NC2COCC2NC(=O)Cc2ccc(C)s2)c(F)cc1F C1(NC(CCCC)=O)CCC2CCN(C(=O)COCc3cc(C)no3)C1C2 N1(C(Cc2c(C)nsc2)=O)CC2(CCN(C(C3CC(Cl)(Cl)C3)=O)C2)C1 C1(OCCC(=O)NCCN(C2CCCC2)C(=O)CC2CC=CCC2)CCCOC1 N1(C(C(=O)OC)C(C)C)C(=O)NCC(c2ccc(O)cc2)C1=O C1(NC(Cn2c(CCC)ncc2)=O)CN(C(=O)CS(=O)(=O)CC)CC1N=[N+]=[N-] N1(C(CCOC(C)=O)=O)C2CCC1CC(F)(CNC(=O)CC1CCCO1)C2 N1(C(C=CCC)=O)CCC2C(CCN2C(=O)C=CCN2CCCCC2)C1 CCS(=O)(=O)c1ccc(OC)c(NS(=O)(=O)c2cc(OC)c(OC)c(C)c2)c1 C1(CC(=O)NCCCCN(C(C(N2CCOC2=O)C)=O)C)CSCCS1 C1(C)(CC)CC(NC(=O)CC(C)(C)CN(C)C)CN1C(=O)Cc1cc(CO)on1 O(NC(=O)C(CCSC)NC(=O)C(O)CC(C)C)CC=CC CCCC(C(=O)NC(CNC(c1ncncc1Br)=O)CC)OC C1(CC(=O)N(C)CC2CCN(C(=O)CCc3cn(C)cn3)C2)CCCS(=O)(=O)C1 C12(NC(C(C)(C)OCC)=O)CC(C1)N(C(c1cc(COC)[nH]n1)=O)C2 C1(c2nc(C(=O)OC)c(C)s2)CCCN1N1CCC(N2CC(=O)NC2=O)CC1 C1(C(N2C(C)CCC2C)=O)CC2(CC(NC(c3ccccc3Br)=O)C2)C1 C(=O)(C(CO)N(C(=O)CN(C1CCC1)C)CC)N(C(CC)C)CCO C=CC(CCC)CC(=O)N(C1CCN(C(=O)Cc2ccc(OCC)nc2)C1)CC C1(NC(c2c(C)nc(C(C)(C)C)s2)=O)CCCN(C(=O)Cc2ccsc2C)C1C c1(C(C)NC(=O)C(c2cccc(C(F)(F)F)c2)N)cc(F)ccc1N(C)C c1(C(=O)NCC(CC(C)C)NC(=O)Cn2ncnn2)ccn2c1CSCC2 c1(C(N2CCC(COC)(NC(=O)C(C)C(C)C)C2)=O)ccncc1N=[N+]=[N-] O(NC(=O)CC(C)(C)NC(c1ccc(N)c(F)n1)=O)CC=C Cc1ccc(C(N2CCCCC2C(=O)NC2(c3ccnn3C)CC2)=O)cc1F c1(C(N2CC(NC(C(C)OCC=C)=O)C(C)(C)C2)=O)n[nH]c2c(OC)cccc12 C12(C(=O)NCC3(CNC(C(CC=C)(C)O)=O)CCC3)CC1COC21CCC1 O=C(CC1CCOc2ccccc21)NCC1(NC(C2CCS2(=O)=O)=O)CCCC1 N1(C(CC2(C)CC2(Cl)Cl)=O)CCN(C(=O)COc2ccccc2)CC1CO c1(CCC(N2CCC(NC(C(C)(C3(C)CC3)OC)=O)C2)=O)cc(C)nc(C)c1 N#CC1=C(C(=O)NCC2(CNC(=O)C(Cl)=CCl)CCOCC2)CCC1 C1(c2n(CCc3ccc(C)cc3)nc(CO)n2)Cc2ccccc2C1 Cc1ncc(CCC(=O)NCC2CCN(C(=O)Cc3cnn(C)n3)C2)s1 C(=O)(CC(C(F)(F)F)c1cccc(F)c1)NC(CNC(c1c(C)scn1)=O)CO C(C1CN(C(C2CN3CCC2C3)=O)CC1C(=O)NC(C)(C)COCC)=CC c1(C(N(CC(N2CCN(C)C(CO)C2)=O)CC2CC2)=O)cnn2ccccc12 c1(C(=O)NCC(CC)(C)NC(c2cn3ccccc3n2)=O)ccc(S(C)=O)cc1 CCC(C#N)C(=O)NCc1ccc(C(N2CC(CNC(N)=O)C2)=O)cc1 N1(C(C(C)NC(=O)NCC)=O)CC2CC2(CNC(=O)C(C)(C)OC(C)C)C1.OC N1(C(Cc2ccn(C)n2)=O)CCCC(n2cc(CCNC=O)nn2)CC1 CC(C)C(F)(CNC(C1(C)CNC(=O)C1)=O)C(=O)N1CCC2CC12 C(C(=O)NNC(=O)C1CCOC1C(C)(C)C)C1(OCC)CCCC1 c1(C(S(=O)(=O)CC2CC2Cc2ccccc2)C)cc2ccc(Br)cc2s1 c1(C(N2C(CNC(=O)CCc3cnoc3)CC2)=O)cccc2[nH]ccc12 C(C(C(=O)N1CCC(c2nc[nH]n2)C1)NC(=O)CCc1cnco1)N(C)C C1(NC(C(C)OC2CCOC2)=O)C2CCCN(C(C3OCCCO3)=O)C2C1(C)C CC1(C(=O)NCC2CCCCN(C(=O)CSC(F)F)C2)CC2CCC1C2 c1(NCCCCCN(C)C(C2CC(=O)NC(=O)C2)=O)ncc2ccccc2n1 Nc1cc(C(=O)NC2CCN(C(C3CCCOC3)=O)C2)ncc1F c1(NC(=O)NC(C#CCC)(C)C)nc2ccc(N)cc2s1 c1(C(CF)NC(C(=O)NCC(C)(CSC)OC)=O)ccc(Br)cc1 c1(C(C)SC(C)(C)C)nc(C2CCC2)ncc1Br C(=O)(N=c1nc(SC)[nH]s1)NCC.c12ccc(cc1)ONC2=O C1(N(C(c2c(OC)cc(C)s2)=O)C)CN(C(c2cccc(F)c2N)=O)CC1(C)C N1(CC(=O)NCCC2CCCCN2)CCCCC1CCO CC1(CC(=O)NC2CC(NC(=O)NC3CCOC3)C2)CCC2(CC1)OCCO2 C1(C(=O)NCC2(C(=O)NC3(C(=O)OC)CC3)CC2)CC1(F)F C(C(C)(C)C(=O)N1CCCC(CN(C(=O)CC2(OC)CC2)C)C1)OC N1(C(C(CC)(C)O)=O)CCC2(CCC(CNC(C3CC4(CC4)C3)=O)O2)CC1 c1(C(C)C)nc(C(=O)N(CCCNC(C2=NC=S2c2ccccc2)=O)C)co1 c1(OCCC)ccc(CN2CCOCC2CC(=O)NCc2cncs2)cc1 C(=O)(CCCCN(C)C(C)C)NCC1(O)CC(NC(C2CN(CC(C)C)C2)=O)C1 c1(C(=O)NC2CN(C(=O)CCC3CCCC3)C2)ccccc1-c1ccccc1 CCC(CN(C)C)C(=O)NC(C)C(=O)N(CC)Cc1cccnc1 c1(C(=O)NCCNC(Cn2c(C)ccn2)=O)coc2c1C(O)CCC2 N1(CC(C)(C)F)C(=O)CCN(C2CCc3ccccc32)CC1=O C1(C(N2CC(C)OC(C)C2)c2nnnn2C(C)(C)C)(COC)CC2CCC1CC2 CCC(C#N)C(=O)NC(C)CNC(=O)CCCc1cnn[nH]1 Cc1nn(CC(C)C)c(C)c1CC(=O)NC(C)CNC(C1(C#N)CCCCC1)=O N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC(NC(c2ccnnc2)=O)C12CCC2 C(=O)(C(C)(C)C(F)F)N1CC(C(C)NC(CCOCCOC)=O)C1 c1(C(N(CC(CNC(C2(COC)CC=CCC2)=O)(C)C)C)=O)cc(C)cc(C)c1 C(=O)(CC(O)C(C)CC)NCC(CC(=O)NC1CCN(CC)C1=O)C1CCC1 C(=O)(CC(CCCC(C)C)NC(c1cccc(OC)c1Br)=O)OC C(CCCCC1CC1)(C(=O)NCCOCC1CC1)N1C(C(=O)NC)CCC1 c1(C(=O)NC2CCCN(C(C3(COCC)CC3)=O)C2)cc(Cl)c(OC)cc1C CCCC(CNC(C1CN(C)CCN1C(C1CCCC1OC)=O)=O)CCO CN1CCC(=CC(=O)N(CCCCNC(=O)C=Cc2cnn(C)c2)C2CC2)CC1 C1(NC(c2c(C)[nH]cc2)=O)CCC2CN(C(C3CC4(C3)CC4(F)F)=O)CCC2C1 C(=O)(C(C#N)C(C)(C)C)NCCCC(C)(C)NC(=O)C1=COCC1 CC(C)C(CCc1ccccc1)C(=O)NC(CNC(=O)CNS(N)(=O)=O)C1CC1 C(=O)(C1COc2ccc(Cl)cc21)N1C(C)CC(NC(c2cnoc2)=O)CC1 N1(C(=O)OC)CCOCC1C(=O)N(CC(=O)NC1CN(C(=O)CC(C)(C)C)C1)C CCC(C)C(O)C(C)C(=O)NCC1CC(C(=O)NC2CC(O)CC2O)=NO1 N1(C(C(CO)OC)=O)CC=CC(C(=O)NCCC2CCCN(C)C2)C1 C=C(C)CC(C(=O)NC1COCC(C)(C)C1)NC(C1C(=C)C1C(=O)OC)=O CC(C(=O)N(C1CCCN(C(c2ccc(CS(C)(=O)=O)cc2)=O)C1)C)S(N)(=O)=O C(c1ccc(OCC(N)=O)c(OC)c1)=CC(=O)N(C)CCN(C(=O)CC#N)C N1(C(c2n(CC=C)ccc2)=O)CC2(CCC(CNC(C3CCC4CC34)=O)O2)C1 c1(OC)ccc(C(N2CCCC(O)(CN(S(=O)(=O)C3CC3)CC(N)=O)C2)=O)c(F)c1 N1(C(c2scc(C#N)c2)=O)CC2CCC1CN2C(C1C2CCCC12)=O N1(C(C(C)OCC=C)=O)CC(NC(c2csc(S)n2)=O)C(C2CC2)C1 C(=O)(C1=Cc2ccc(F)cc2OC1)NCCC1N(C(CSCCC)=O)CCSC1 n1(CC(=O)NCCCN(C)C(c2cnc(S)n2C)=O)nc2n(c(=O)c1=O)CCC2 c1(CNC(C2C(NC(c3cccc(COC)c3)=O)C2)=O)ccc(F)c(C#N)c1 Cc1cnc(NCC2CCCN(C(=O)CCSC3CCCC3)C2)c([N+](=O)[O-])c1 CC(C)CCC=CC(N1CCC(NC(C2(Cl)CC2(F)F)=O)C1)=O N1(C(c2ccc(C)nc2C)=O)CC(NC(C2CC(C)(O)C2)=O)C(S(C)(=O)=O)C1 C1(C(N2CC(CCNC(C3(C(C)C)CCC3)=O)(OC)C2)=O)COC2(CCC2)C1 c1(NC(C2N(Cc3c(Cl)cc(C)cc3Cl)CC2)=O)cc(S(C)(=O)=O)ccn1 C(=O)(CCCC(C)(c1nnnn1C)NC(c1ccc(C(C)(C)O)cc1)C)OC CCCCC(C)C(=O)NC1C=CCN(C(=O)CCC(=O)N2CCC(O)CC2)C1 C(CC(C)(C)C)N(C1CC(F)(F)C1)C(=O)NC(C1CC1(C)C)CC [N-]=[N+]=Nc1cncc(C(N2CC3(CC(NC(c4cc([N+](=O)[O-])c[nH]4)=O)C3)C2)=O)c1 c1(C(=O)NC(CC(C)C)CNC(=O)C=CCn2cncn2)ccn(C)c(=O)c1 N1(C(C2C(OC(C)=O)CNC(=O)C2)=O)CCC2(CC1)CN(C(=O)N(C)C)CC2CO c1(CN(C(=O)C(N2CCC(CO)(OC)C2)=O)CC=C)ccc(C(F)(F)F)c(Cl)c1 Cc1ccnc(C(=O)NCCOCCCNC(=O)CC2CCCCCC2)c1 c1(OC)ccc(C=CC(C)NC(c2nc(C3CCNCC3)co2)=O)cc1OC C(CC(=O)NC1(CNC(c2oc(C)cc2C)=O)CC1)(C1=CCCC1)OCC C1(N(C(c2nc(COC)oc2)=O)C)C2CN(C(c3ccc(Cl)cn3)=O)CC12 C1(C(N(CC)CC)=O)CCCN(C(c2ccc(F)c(Br)n2)C(=O)NC2CC2)CC1 C1(C(N2CC(C(=O)Nc3cnn(CC(F)F)c3)C2)=O)CCC2(CC1)CC2 C1(C(C#C)C)CCN(C(N2CCC(OC(C)(C)C)C2)=O)CC1 C(=O)(C1=CCS(=O)(=O)C1)NC1CC(N(C(c2ccc(C)nc2)=O)C)C1 N1(C(CC2(CSC)CC2)=O)CCC(O)(C(C)NC(c2cccc(C)c2)=O)C1 N#CC1(C(=O)NC2CCN(C(=O)C=CC(N)=O)CCC2(F)F)CC2CCC1CC2 Cc1ccc(C(N2C3CN(C(=O)C(C)(C)c4ccccc4)CC23)=O)cc1Cl Cc1cc2cccc(CN3CCN(C(=O)Nc4ccn(C(C)C)n4)CC3)c2[nH]1 C(C(C)(C)C1=CCCC1)N.C12(C(=O)OC)CCC(NC(=O)CCCC3CC3C)(CC1)C2 N1(C(C(C)Oc2cccc(C)c2)=O)CCC(NC(C2CC2C)=O)C12CC2 N(C(=NCCF)NCC1(O)CS(=O)(=O)C1)C(c1noc(C)n1)CC c12ccc(cc1)[nH]2.CC(O)CC(=O)N(CC(C)NC(C1CCCO1)=O)C N1(C(C2CCN(CC)CC2)=O)CCC(NC(=O)CCSC)C(CO)C1 N12CCC(CC1)NC(=O)C2C.C1(CNC(CSC)=O)CCCCC1OCCOC C12(CCNC(C(C)(C)n3cccn3)=O)CCC1CN(C(C1(C(F)F)CC1)=O)C2 C1(C)(NC(CC(C)N(C(=O)CC2NC(=O)NC2=O)C)=O)CCC(C)C1 C(=O)(C(CC1CCOCC1)NC(C1CC(F)(CF)C1)=O)NCC1CC(=C)C1 c1(CC)cccc(C(=O)NC2CC(NC(C34CCC3C4)=O)C(O)C2)c1O n1(CCC(N2CC3(C2)CC(=O)N3)=O)cnc([N+](=O)[O-])c1.C1(C(C)(C)C)C=CCC1 CN1CC(O)CC1C(=O)NCC1CC(NC(=O)CCCSC(C)(C)C)C1(C)C CCCC(C(=O)NC1(COC)CN(C(=O)CCc2ccoc2)C1)c1ccccc1 N1(C(c2cnc(C#N)s2)=O)CC2(COC(CNC(=O)C(CO)NC(N)=O)C2)C1 CN1CCOC(C(=O)NC2CC(CNC(=O)CS(N)(=O)=O)CC2O)C1 C1(NC(c2c(C)ccnc2)=O)CC2(CCC(CNC(c3cnc(O)s3)=O)CC2)C1 c1(OC)cc(C(=O)NCC(c2ccccc2)N(C)C(C2CC2C)=O)cc(Cl)c1 CC#CCC(C(=O)N(C)CC1CC1C)NC(=O)CCC(C)CC Cc1c(-c2nc(Cc3cccnc3)nn2CC(C)CO)cnc2ccnn12 CCCC(C(=O)NC1CC(NC(c2cc(CC)cnc2O)=O)C1)NC(C)=O C1(NC(C(=O)Nc2ccc(C(=O)NC)cc2)=O)CCc2cnn(C(C)C)c2C1 N1(C(C(CC#C)C2CC2)=O)CCOCCC1C(=O)NCC(c1cccs1)C CC(CF)CC(=O)NCCCCNC(c1nc(C(F)(F)F)cn1C)=O Cc1nc(O)nc(C)c1CC(=O)NCC(CNC(C1(Cl)CCC1)=O)CO c1(N(c2ncc(Cl)cc2O)C(C2CCNC2)=O)ncnc2cc(F)ccc12 C1(n2cc(C(CCC=C(C)C)NC(=O)CC(=O)NC)nn2)CCCC1CCC N1(C(CCOC)=O)CCCC(CCNC(c2cc(SC)oc2C)=O)CC1 C(C(=O)N(C)OC1CCCC1)(C1CCCC1)NC(C1C(C(C)C)C1)=O N1(C(CC2(NC(CC(C(=C)C)OCC)=O)CC2)=O)CC2(CCC(=O)O2)C1 CN1CCC(C(=O)NCCC2(C)CCN(C(c3ccc[n+]([O-])c3)=O)C2)CC1=O CCCC(C)(C)C(=O)NCC1CN(C(=O)C(CCOC)OC)CCCO1 N1(C(C(C2CCC2)NC(Cc2cc(C)nn2C)=O)=O)CC(=O)N(C)CC1C C(C(N=[N+]=[N-])C(=O)NC1CCC(NC(c2n[nH]cc2C2CCC2)=O)C1)OCC C1(NC(=O)NC2CCC(CC#N)C2)CC2CC1CC2F C1(COC)CN(C(=O)CNC(C2COC2)=O)CCN1C(C1CCCCC1)=O C(C)(C)(C(C)CC(=O)NCCc1c[nH]nc1O)NC(c1ccn(COC)n1)=O c1(C(N2C(CCNC(c3cncc(N)n3)=O)CCCC2)=O)cc(F)c(F)cc1F C(C)(C(CC(=O)NC12CC(F)(C1)C2)NC(c1cc(N)cc(F)c1)=O)OC C(CCCCCNC(C1CC2CC1C2)=O)NC(c1cscc1Br)=O C(=O)(CCCCC#Cc1ccccc1)NC1CCN(C(C2C(=O)OCC2)=O)CC1 c1(CCCNC(=O)C(N2CCN(c3cccc(Cl)n3)CC2)=O)ccc(O)cc1 C1(CNC(C2(CC#C)CCCO2)=O)C2CN(C(C3CC4(CC4)CO3)=O)CC12 c1(N(CC(C)C)C)cccc(NC(=O)N(CCCOCC(F)(F)F)C)c1 c1(CCC(=O)NCC2CN(C(CCC#C)=O)C2)ccc(F)c(F)c1 C1(OCC(C)C)CCN(C(=O)CC23CCC2CN(C(=O)CC(=O)NC)C3)C(C)C1 Nc1cc([N+](=O)[O-])ccc1C(=O)NCC1CN(C(C2CCSC2)=O)CCO1 S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)N(C)Cc1cncs1 CS(C)(=O)=NC(=O)c1cc(C2COC2)on1 N1(C(C2N(CC)CC2)=O)CCCCC(N(C(=O)Cn2cncn2)C)C1 C1(NC(C2CCC(C)C2)=O)CC1C1CCCN(C(c2ccc3scnc3c2)=O)C1 N1(C(C(C=C)C)=O)CCSCC1C(=O)NCC1CCCCN1C N(C(=NCCC1CC=CC1)NC(c1cccc(F)c1)C)C(C=C)C N1(C(C(=O)Nc2c(C)cccc2)C2CCC2)CCC(O)(CN(C)C)CC1 c1(CC(=O)NCC(C)(C)NC(c2cc(F)cc(N)c2F)=O)ccn2cncc2c1 c1(NC(C)=O)ccc(C(=O)NC(C)Cc2cccc(C(C)(C)C)c2)nc1 N12CCN(CC1C1CC1)CC2=O.C12(CN(C3CC3)CC)CCCC1C2(F)F c1(C(c2n(CCC)nnn2)Nc2ccc(C)nc2)ccc(C(C)CC)cc1 Cc1ncn2ccc(C(=O)NCC3(CCNC(=O)C=Cc4cccs4)CC3)cc12 Cc1cc(C(=O)NCCN(C(c2ccn3ccsc23)=O)C2CC2)c2nccn2c1 N1(C(COCCNC(=O)CC2CNC(=O)O2)=O)C2C=CCC1CC2 C1(O)(CCNC(C(C)(C)C2CCCC2)=O)CCN(C(C2C=CCCC2)=O)C1 C(c1ccccc1)=C(CC)C(=O)OC(C)C(=O)C1CCC1 c1(NC(C2C(C(=O)Nc3c(C#N)cno3)C2)=O)ccc(F)c(F)c1O c1(C(=O)NCCN(C(=O)CC(C)C(C)C)CCOC)cccc(F)c1O C1(C)(CNC(C(CC)(C)CC)=O)CC(F)(F)CN1C(=O)Cc1ccc(C)c(F)c1 c1(C(N(CCNC(C=CCC)=O)CC)=O)cc(C)cc(Br)c1F.C(C)(C)(CC)O c1(N2CCC(C)(C(=O)NC)C2)ccc(S(=O)(=O)NCc2c[nH]c(=N)s2)c(Cl)c1 CN1C(=O)NC(C2CCN(CC(=O)Nc3ccc(=N)[nH]c3)CC2)C1=O C1(CC(=O)NCc2ccc(CNC(C3(CO)COC3)=O)cc2)CC2CCC1C2 CC1CCCc2nc(C(N3CCOC(CCNC(=O)C(C)(C)C#N)C3)=O)cn21 c1(C(N(CCCCC)CCC(=O)NCCC(=O)OCC)C)cnc(C)[nH]1.C1CS1 CC1CCN(C(C2CC(=O)N2)=O)CC1CNC(=O)C(c1ccc(F)cc1)F C1C(C)(CC(C)C)O1.c1(C(=O)NCCOCCOCCC)cc(OC)ccn1 c1(OC)nc(N2CCC(C)(NC(C3CCC3(C)C)=O)CC2)nc(C)c1F C(=O)(CCC(C)(C)F)NC(COC)C(=O)NCc1ccc(O)c(C)c1 Cn1nc(C(=O)NCC2CC2NC(c2sccc2Br)=O)cc1C(N)=O C(c1nc2ccccc2o1)=CC(N1CC(C)N(C(=O)Cn2cccc2)CC1)=O c1(CC(=O)NCC2CC(NC(C3C(CN(C)C)C3)=O)C2)cccc(Cl)c1Cl CC1(CNC(=O)COc2ccc(F)cc2F)CN(C(C2(C)CC2(Cl)Cl)=O)CCO1 Cc1ccc2c(c1)CC(C(=O)NCC1CCCCN1C(C1CCCCCC1)=O)O2 C#CC(CNC(=O)C(C1CCCO1)NC(=O)Cc1sccc1C)CC(C)(C)C c1(NC(C(CNC(c2ccc(CC)[nH]2)=O)O)=O)ccnc(OC)c1 N1(C(c2c(CC)nccc2)=O)CCC2CC2(C(=O)NC2(C)CCSCC2)CC1 C12(NC(c3[nH]cc(CC)c3)=O)CCCCC1CN(C(c1nocc1Cl)=O)C2 N1(CC(=O)NC)CC=C(CCNC(c2cc3c([nH]2)CCCC3)=O)CC1 c1(C(=O)NC(C)CCNC(=O)CC(F)(F)Cl)cc2cn[nH]c2cn1 c1(C(=O)NCCCC2(NC(CC3(C)CC3)=O)CC2)cc2n(n1)CCCO2 C1(CNC(C=CC(C)(C)C)=O)CCCCN1C(c1ccc(-n2ccnn2)cc1)=O c1(NC(C2C(C(=O)Nc3c(OC)ncnc3OC)C2)=O)cccc2nc[nH]c12 C12(NC(C(C)NC(CC)=O)=O)CCCC1N(C(C1CCCC3CC13)=O)CCC2 c1(C(=O)NC2CCCC(NC(C(N)=O)=O)C2)nc(Br)c2ccccn12 c1(C(=O)NC2(C)CCCN(C(c3cc(C(C)=O)oc3)=O)C2)nc2c(s1)COCC2 C(C(=O)N(C)Cc1ccc(C)nc1)(C(C)CC)NC(c1ccc(CC)cc1)=O c1(N2CCC(CCCC)C2)nc(N2CCC(CC(F)(F)F)C2)cc(C)n1 C=CC(C)(CC)C(=O)NCC(C)(CO)NC(=O)COc1ccsn1 CC1CCCC1N=c1nc(N2CCC(C)(N3CCC3)CC2)c2ccccc2[nH]1 c1(C(=O)NC(c2cccc(C)c2)CNC(C(CC)F)=O)ccc(C2CC2)nc1O c1(OC)ccc(C(O)CNc2ccc(C(=O)NC3COC(=O)N3)cn2)cc1 C1(F)(CNC(c2cc(C(F)F)ccn2)=O)CCN(C(c2ccnc(S)c2)=O)C1 CCCC(O)CC(=O)NC1CCCC1NC(c1cn(CCC2CC2)nn1)=O C1(CC=C)COCC1NC(=O)CCCN(C(=O)C(C)OCC1CC1)C C1(NC(C=CCC)=O)CC2CN(C(c3cc[nH]c3C(C)C)=O)CC12 CC1CC(N=c2[nH]c(=NCC3CCC3)c3cc(F)cc(F)c3[nH]2)CCS1(=O)=O C#CC1(C(=O)Nc2cccc(OC)c2C)CCN(C(=O)CC2CC(CC)=NO2)C1 CCCC(CC)C(=O)N(CCCOCCN(C)C(c1cnc(C(F)F)s1)=O)C N1(C(c2ccc(Br)cc2[N+](=O)[O-])=O)CCC2(CC1)OCCC2O N1(C(c2c(OC)ccc(C)n2)=O)CC2CS(=O)(=O)CC2(NC(=O)C(F)F)C1 c1(N)cc2scnc2[nH]1.C1(C(=O)NCCCOCCNC(=O)OCC)CC1(C)Br C1(COC)(NC(c2cc(CO)[nH]n2)=O)CN(C(=O)CCc2ccc(Cl)s2)C1 Cc1cc(C(F)F)oc1C(=O)NCC(CO)NC(=O)Cc1cnccn1 c1(CNC(C2(SC)CC2)=O)ccc2c(c1)CCN(C(C1CC3CCC3C1)=O)C2 c1(OC)ncc(-c2ccc(N3CCN(Cc4ccc(C#N)s4)CC3)cc2)cc1C N1(CCCC(N2CC(CN)C(F)(F)CC2)=O)C(=O)Cc2ccccc2C1=O N1(C(C(C(C)C)CNC(=O)CC(C)n2ccnc2)=O)CC2(C)CCC2(C)C1 N1(C(CSc2c(C)cccc2C)=O)CCC2(CC1)CC2NC(c1cnsn1)=O C1(O)(C(C)NC(CC(C)C)=O)CCN(C(c2cc(Br)co2)=O)C1 O=C(NOCC=CCl)C1c2c[nH]nc2CN1C(=O)C1=CC2C=CC1C2 CC(C)C(C#N)C(=O)N(C(C)CCNC(c1cccc(F)c1Br)=O)C C1(O)(CN(C(=O)Cn2cnnc2)C)CCN(C(=O)Cn2cc(Cl)cn2)C1 CC(C)CC(CNC(C12CCC(C)(C1)OC2)=O)C(=O)NC1CCCC12CC2 CC1COC(C(=O)NCC=CCNC(=O)C=C2CCOCC2)C1 C1(CNC(=O)NC(c2cccc(OC(F)(F)F)c2)CO)CC2CCCC2O1 n1(CC(=O)NC(CNC(Cn2c(C)ccn2)=O)C(C)C)cc(Cl)c(C)n1 c1(C(C(=O)NC(CC)(C)C)N(C2CCCC2C#N)C)ccncc1CC c1(C2CCN(C(=O)NCC3(COC)CC3)C2)nc2ccccc2o1 C(=O)(CC1=CCCCC1)N1CC2C(CNC(COc3c(C)c(F)ccc3)=O)C2C1 c1(C(=O)NCC2C(NC(C(CSC)C)=O)CC2)nc(C2CC2)ncc1Cl CC1(C)C2CCC1(C(=O)NCCNC(C1CCc3ncnn3C1)=O)CC2 C(C(C(=O)NCC1COCC1NC(C1CC(Cl)(Cl)C1)=O)N(C)C)OC c1(-c2c(C)csc2)nnc2n1CCCN(C(c1cc(I)ccc1F)=O)C2 c1(OC)nccc(C(N2C(C(=O)NC3CN(C)C3)CC3CC23)=O)c1Cl c1(C(=O)NC2CCC(CNC(C(CC)F)=O)C2)ccnc2[nH]c(CC3CC3)nc12 N1(C(C2(CC)CC2(F)F)=O)CCN(C(=O)Cc2cc(C(C)C)no2)CC1C c1(C(=O)NCC2CC(CNC(C(CC=CC)C)=O)C2)c(O)nnc2c1COCC2 n1(CC)cc(Cl)cc1C(=O)N(CCN(C)C(c1sc(OC)nc1Cl)=O)C(C)C C1(C(N(CC(C)(C)NC(=O)CN2CCCCC2)C)=O)CC12CCC1(CC1)CC2 C1(NC(=O)CN2CCC(O)CC2)CC2CN(C(=O)Cc3cc[nH]n3)CCN2C1=O C(=O)(C(C)(C)C(F)(F)F)N1CC2(C(C(=O)Nc3c(C(N(C)C)=O)cccc3)C2)C1 C1(CCNC(C(N2CCOC2=O)C)=O)CCCN1C(=O)CCSC(F)(F)F N1(C(CC2C(=O)NC(=O)N2)=O)CC2CCC1CN2C(c1nccc(Cl)c1O)=O N(C1CCCNc2ccccc21)C(C1COCCN(Cc2c(OC)ccs2)C1)=O c1(C(=O)NCC2(F)CC(NC(=O)C=CCO)C2)ncnc2ccsc12 CCC(CNC(C1(CCOC)CCC1)=O)(CC)NC(=O)C(c1ccc(C)cc1)C Cn1c(C(=O)NCC(F)CNC(=O)C(C2CCCCC2)F)cc2ccc(O)cc12 N1(C(c2ccc3c(c2)COC3)=O)CCC2(CCN(CCC3CCCCC3)CC2)C1 CN1CCC(C(N2CCCC2CN=[N+]=[N-])=O)(NC(=O)C=Cc2ccncc2)C1 c1(OC)ccccc1CC(=O)NC1CCC1C(=O)NC1CCC(C(N)=O)C1 c1(OC)cc(C)c(C(=O)NCC23CC(CNC(=O)C(C)CSC)(CO2)C3)cn1 c12ccoc1C2.c1(C(=O)NCCCOCCNC(C(C)C)=O)cn(CCO)nn1 c1(N(C(C2(C#C)CNC2)=O)CC2CCCC2)cc(C(F)(F)F)ccn1 c1(C(N2C3CN(C(CCC(CC)OC)=O)C(C3)CC2)=O)cc2ccnc(Cl)c2s1 c1(NC(CCNCCCN)=O)ccc(Br)c2c1OCCC2 N1(C(c2nnc(C)s2)=O)CCC2(CC1)CCN(CCC1CC1)C2 Cc1cc(C(C)(C)C(=O)NCC(C)NC(=O)CC(O)c2cnc(Cl)s2)cs1 CC1Cc2ccc(F)cc2C1NC(=O)Cc1c[nH]c2ccccc12 c1(N2CC3(C(NC(C(C4CC4)OC)=O)CCS3)C2)cc2nnc(C(C)C)n2cn1 c1(CCN)ccc(C(C(C(CC)C)C)c2nnnn2CCOCC2CC2)cc1.OC c1(C(=O)NCC(CC)(C)NC(=O)C=C(C)C)cn2c(C)cccc2n1 C12(C(=O)NC3CCC(CNC(C4C(=C)C4)=O)CC3)C3C4C1C1C2C3C41C c1(NC(CCCC)c2nnnn2CC2CCOC2)ccc(SC)cc1 C(=O)(C1=CCCOCC1)NC1(CC)CCCN(C(c2cc3n(n2)CCCC3)=O)C1 C1(CCNC(CSCCC)=O)C(C)CCCN1C(c1scnc1C)=O Cc1nccc(Cl)c1C(N1CC2C(CNC(c3sc(=N)[nH]c3C)=O)C2C1)=O C1(C(=O)NCc2snc(CC)n2)CCC2(CC2)N1C(C12CCC(OC)C1C2)=O C1(C(=O)NC(CCSC)CO)CC(=O)CN1C(C1CC1[N+](=O)[O-])=O C1(NC(c2cc(CC)[nH]n2)=O)CC2CC(NC(c3cscc3C(F)(F)F)=O)C1C2 c1(N2CCCN(C(CC#N)=O)CC2)ccc(S(=O)(=O)NC(=O)C2CC2)cc1[N+](=O)[O-] C(=O)(CCC(F)(F)F)NC(C(=O)NCC(CO)N(C)C)CCF Cc1cccc(Br)c1C(C(=O)N(C)CCC1CCCO1)NC(C1CC1Cl)=O c1(C(=O)NCC2C(NC(C(CCC)OC)=O)C2)cc(Cl)ccc1C N1(C(C2C(C)=C2)=O)C2CCC1C(C)C(NC(c1nc(C(F)(F)F)cn1C)=O)C2 CCC(CC)(CC)C(=O)N1CC(NC(c2cnnc(C)c2)=O)C(C2CC2)C1 C1(CC)CCCN(C(c2ccn(C)n2)=O)C1C(=O)NCCC(C)O Cc1cc(C)cc(S(=O)(=O)NC2CC2C(=O)Nc2cnn(C(C)C)c2)c1 C1(C2CCN(C(=O)Cc3cccc(O)c3)C2)(NC(CC2C(C)=NOC2=O)=O)CC1 C(CCN=c1[nH]c2ccc(O)cc2s1)N(C(c1ccc(S(C)(=O)=O)[nH]1)=O)C1CC1 c1(CC)ccc(NC(=O)NC2CC(NC(c3ccnc(C)c3)=O)C2)cc1Cl c1(C(N2C(C(CNC(C3C(C)C3)=O)O)CCCC2)=O)cc2c(cn1)COCC2 Cc1cc(C(=O)NC(CNC(=O)C=Cc2nccs2)C2CC2)cc(C)n1 C1(n2cc(CCSCC)nn2)CCC(C(=O)NC(N2CCN(C)CC2)=O)CC1 C1(F)(C(=O)NCCN(C(c2cnc(O)c(F)c2)=O)CC)CCCN(C)C1 N1(C(C2N(C(c3ccnnc3)=O)CC(=O)NC2)=O)CC2CCC1C(O)C2O C=C(CNC(=O)C(OC)OC)CCNC(c1[nH]nnc1C(F)F)=O Cn1nc2cccc(C(N3CC4CCC3CN4C(=O)Cc3nnc(O)s3)=O)c2n1 N1(C(C(C2CCN(C(C(CCC)F)=O)CC2)C)=O)CCCC(O)CC1 C1(Cc2cn(CCNC(C(c3ccccc3Cl)(C)C)=O)nn2)CC(F)(F)CO1 c1(C(N2C(C(=O)Nc3ccccn3)CC3CC32)=O)c(F)cncc1Br c1(N(C(CC)C)C)cc(N(C)CCOCCOC)nc(COC)n1 c1(C(=O)NC(CNC(c2ncccc2Br)=O)C2CC2)ccc2c(c1)CC2 C1(NC(COC2(C)CCCC2)=O)CN(C(C2CCCOC2)=O)Cc2ccnn2C1 c1(OC)ncnc(OC)c1C(=O)NCC(C)NC(c1sccc1C#N)=O C(C(CC(F)(F)F)NC(C1CC1C1CCC1)=O)NC(=O)Cn1ccc(C2CC2)n1 c1(C(N2CCC(NC(c3c(C)noc3N)=O)C(F)C2)=O)cccc2occc12 CC(C)CC(CNC(=O)COOCC1CCCO1)NC(c1n[nH]c(C(C)C)n1)=O N1(C(CC=CC)=O)CC(CNC(c2cnn(CC)c2)=O)C(F)(F)C1 C1(C(=O)NCc2cc(C)nn2C)COC2(C1)CN(C(=O)C1=C(C#N)CCC1)C2 Cn1ccc(=O)c(C(=O)NC2COCCN(C(=O)CCC3CC(F)(F)C3)C2)c1 Cc1cc(F)cc(C)c1C(N1CC(NC(=O)C(C)CC(C)C)C(C#N)C1)=O CCCC(C(=O)OC)OCOc1ccc(CC(=O)OCC)cc1 C1(NC(C(c2nc(C)sc2)=O)=O)CN(C(C2(N3CCCCC3)CCC2)=O)CC1O CCC(C)N=C(NC1CC(N(C)C(=O)OC(C)(C)C)C1)NCC(F)F c1(C(N2CC(C)(NC(c3cc(C#N)ccn3)=O)C2)=O)ccnc2c1CC(=O)N2 c1(OCC2CC2)cc(C(N2CCC(N(C)C(C34COCC3C4)=O)C2)=O)ccn1 N1(C(c2ccc(OC)s2)=O)CCC2CC2(NC(c2sc(=N)[nH]c2C)=O)CC1 C1(NC(=O)CC2CCCCCC2(F)F)CN2CCC1c1ccccc12 CCCC(C(=O)NC(C1(O)CN(C(=O)CNS(N)(=O)=O)C1)C)N(C)C C#Cc1ccc(C(N2CC(NC(c3sc(Cl)cc3Br)=O)CC2C)=O)o1 c1(C(N2C(CC(=O)NCC3C(C)NC(=O)CC3)CC2)=O)cnn2ccccc12 C1(NC(c2c(C)cnc(Cl)c2)=O)CCN(Cc2cccc3[nH]ncc23)CC1(C)C C1(C(=O)NC2CCC(NC(c3ccc(C(F)F)o3)=O)CC2)CCN2CCCC2C1 C1(CC=C)(NC(c2cnncc2NC)=O)CCN(C(=O)C(F)C(C)C)C1 N1(C(C(C)(N(C(=O)Cc2cc[nH]n2)C)C2CC2)=O)CCC(C(N)=O)C1 N1(C(CC2OCCN(C(CC3(COC)CC3)=O)C2)=O)CCS(=O)C(C)C1 C1(CC(=O)NCC(C(C)C)NC(c2ncsc2C2CC2)=O)CCC(C)(C)CO1 CCCC(O)C(=O)NC1CCN(Cc2nccn2CC)C1 c1(C(=O)NC2CC(NC(C3(CC#C)CCCO3)=O)C2)onc(C)c1C CS(=O)(=O)c1ccc(C(=O)NC2CC2NC(=O)C2=CCS(=O)(=O)C2)nc1 c1(C(=O)NCC(C)N(C(c2cc(CCC)c(C)s2)=O)C)n[nH]c(CC)c1[N+](=O)[O-] N1(CC(=O)NC2CCC(CCNC(c3nc(C(C)C)sc3)=O)C2)CCOCC1=O C1(C(=O)Nc2c(C)nc(N(C)C)cc2)CC2CCC1N(C(=O)C(C)NC=O)C2 c1(CC(=O)NC(C2CN(C(C3CC(C)OC3)=O)C2)C)ccccc1[N+](=O)[O-] c1(C(=O)NCC2C(NC(C(C=C=C)C)=O)COC2)cc(N2CCC2=O)ccc1F C1(NC(C=C(CCC)C)=O)CN(C(=O)CC2CC(C)C2)CC12CC2 c1(C(N2CCC(NC(CCC=C=C)=O)CC2)=O)c(OC)ccnc1OC C(=O)(C1=CC2(CCOC2)C1)NC1CC(NC(Cc2cn(C)nc2Cl)=O)C1 C1(CNC(c2nn(C)c(O)c2)=O)CCCC2(CCN(C(C3CC3C#N)=O)CC2)O1 C1(C(=O)Nc2c(C)ccc(C)c2)CCCN1NC(=O)CC1CC2CCC1C2 N1(C(CN(C)CC)=O)CCCC2CN(C(C3(C4=CCCCCC4)CC3)=O)CC12 C(CN=C(NCC(C)(C)C1CCOC1)NC(C1(C(F)(F)F)CCCCC1)C)SC C1(CN(C)C(c2cnns2)=O)CCCN1C(=O)CCC1CC1(Cl)Cl C(CC(=O)Nc1ccc(CO)o1)(C(F)(F)F)OC.C12CC3CCC(C1)N3C2=O c1(CNC2CCC(NC(c3cc(-c4ccco4)no3)=O)C2)ccnc(Br)c1 c1(OC)cc(C)c(C(N2CCN(C(=O)C(N)=O)CC2)C(=O)NCCSC)c(F)c1 N1(C(C(C)CN(C)C(c2cc(C(C)C)no2)=O)=O)CCCCN(C)CC1 N1(C(CC2(C)CC2(F)F)=O)CCC2(CC1)C(NC(=O)C1CC1)CS2(=O)=O c1(C(=O)NC(C)CNC(C2CC(=O)NC(=O)N2)=O)ccc2c(C)cc(O)nc2c1 C1(CC(=O)NC(c2ccc[nH]2)C)CC(C)N(C(C2OCCC2(C)C)=O)C1 c1(C(=O)NCC2CN(C(Cn3ncc(C#C)c3)=O)CC2C)cc(F)cc(C)c1O C1(NC(CC(CC)C2CC2)=O)C2CC3C(C2)C13C(N1CC(S(C)=O)C1)=O CC(=O)CCCC(=O)N(C)CC1(O)CCCN(C(=O)CCC(=O)c2ccc[nH]2)C1 CN1CC(NC(c2ccc(CNC(=O)CCNC(N)=O)o2)=O)C2(CC2)C1 C1(CC)C(NC(C2CCCS2)=O)CCN1C(=O)CCOc1ccccc1Cl N1(C(c2c(CC)nns2)=O)CCN(C(c2coc(SC)c2)=O)C(C(C)C)C1 C#CCCC(C(=O)NC1CC2CC1CC2=O)NC(=O)CCOCC1CC1 CC1Cc2cc(F)ccc2N(C(C2CC(=O)N(CCN(C)C)C2)=O)C1 C1(C(N2C(C(N(C3(C4CC4)CC3)C)=O)C=CC2)=O)CC2(CCO1)CC2 c1(NCC2(C)CCN(C(CCC=CC)=O)C2)ncnc2cc(OC)c(OC)cc12 CC1(CNC(C2(CC3CC3)CC2)=O)CCC(NC(=O)CCc2cc(Cl)cs2)C1 c1(NCCc2ncc(CO)s2)nc(N2CC=CCC2)nc2scnc12 C(=O)(C(CO)C(F)(F)F)N1CC(OC)C(C(=O)NC2COCC2F)C1 N1(C(CSC)=O)CC(=O)CC1CN(C)C(C1CC(C(F)F)C1)=O Cc1[nH]nc(C(N2CCC(C)(C(=O)NCCc3ccccc3F)C2)=O)c1Cl c1(-c2n(-c3ccc(C)cc3)nc(C3CC3(C)C)n2)cccc(C)c1C C=CCCC(F)(F)C(=O)N1CCCC1CN(C)C(C1CCC(N(C)C)CC1)=O c1(C(N2C(C)CC(CNC(c3cc(C(N)=O)co3)=O)CC2)=O)cc([N+](=O)[O-])n[nH]1 N1(C(Cc2scc(C)c2)=O)CCC(C)C(CNC(=O)CN(C(C2CC=CC2)=O)CC)C1 c1(C(=O)O)cc(CNCc2c(F)cc(I)cc2F)c2ccccn12 O=C1CCC(CCC(=O)NCC2CCN(C(C3(F)CC=CC3)=O)CC2)CN1 c1(C(=O)NCC(C)CNC(=O)CSc2cccnc2)cc2n(n1)CC(F)C2 N1(c2cc(N(C)C)ncn2)CCC2(C1)CN(CC(=O)N=c1cco[nH]1)C2 c1(C(C)C)ncncc1C(=O)NCC(C)N(C)C(C1CCOC1(C)C)=O c1(C(N2CCC(F)(CNC(COCCC)=O)C2)=O)cnc2c(C)cccc2c1 C1(NC(CC(=O)OCC)=O)CCCCN(C(=O)CCc2cscn2)C1 C(c1nc2ccccc2[nH]1)=CC(=O)NCC1CN(C(c2cnc[nH]2)=O)CCO1 Cc1cccnc1C(C(=O)NCCCC1CC1)N(C)C(c1cnn(C)c1)C c1(C(N2CC(CNC(C(CC=CC)C)=O)C(F)(F)C2)=O)c[nH]c2cccc(Cl)c12 O=C1CCCC(C(=O)NC2C=CC(CNC(C3(F)CC3c3ccccc3)=O)C2)O1 C1(CC(N2C(C#C)CCC2)=O)CN(C(c2[nH]nnc2CC)=O)CC12CC2 C1(N(C(C2CCCCO2)=O)CC)CC(=O)N(C2CC2)C1 CCC(C)(C)CCCC(=O)N(CCNC(=O)CC1OCCO1)Cc1ccccc1 Cc1n[nH]c2cc(C(=O)NCCC(C)(C)NC(C3CCCSC3)=O)ncc12 CCC(=O)CCC(=O)NCC(O)C(=O)NCC1COCC1(C)C c1(C(=O)NCC2CN(C(C(COC)OC)=O)C3(C2)CCC3)ccc(C#N)c(C)c1 N1(C(CC(CNC(c2c(C)cc(N)cn2)=O)O)=O)CC(C2=NOC(C)C2)C1 CC(C)C(F)(F)CC(=O)NC1CC(CNC(=O)C(c2cccc(F)c2)(C)O)C1 c1(CNC(c2c(CN)non2)=O)nc2cc(F)c(F)cc2[nH]1 N1(C(C2C(C)CCOC2)=O)CCN(C(c2ccco2)=O)C(c2cccnc2)C1 c1(C(=O)NC2CCCN(Cc3cc(OC)ncc3)C2)ccc([N+](=O)[O-])o1 c1(OC)cc(C(=O)NCC2C(C)CCN2C(=O)CCCC#N)sc1Br C(=O)(C1COc2cc(C)c(C)cc21)NCC(CC)NC(C1CNC(=O)N1)=O C(C)(C(CC(=O)N1CC2C(C(N)=O)C2C1)NC(=O)C(C)c1ccsc1)OC C1(CN(C(=O)Nc2ccc(Cl)cc2)Cc2ccc(F)cc2)CCCC12CCNC2 c1(C(N2C(C)CCC(CNC(C3(OC(C)=O)CC3)=O)C2)=O)ccc2cnsc2c1 C1(NC(=O)CCC2CC2(F)F)CC12CCN(C(C1(CF)CCC1)=O)CC2 Cc1cc(O)ncc1C(=O)NC(CO)CCCCNC(=O)CN(C1CCC1)C c1(C(C)NCc2ccccc2ON)cc(C(F)(F)F)ccc1F.C(C(F)F)OC c1(NC(c2n(C(C(=O)OC)C)nnn2)CC(C)C)ccccc1C(C)(C)C C1(OC)CC(CNC(c2cnc(SC)s2)=O)N(C(c2cccc[n+]2[O-])=O)C1 C1(F)(C(=O)NC(CCN(C)C)(C)C)CCCN(C(C2(CO)CCOC2)=O)C1 c1(C(N2C(CNC(CS(=O)(=O)N(C)C)=O)CCCCC2)=O)cccn2nnnc12 c1(OCCC)cc(C)ccc1C(=O)NCC1C(C(=O)Nc2nccs2)C1 C(CCN=c1[nH]c2c(c(=NC(C)c3nc(=N)[nH][nH]3)[nH]1)CCC2)N(CC(C)C)C Cc1nc(C(C)C)oc1C(=O)NC(C)C(C)(C)NC(c1cnc(=N)[nH]c1)=O c1(C(C)C)ccc(C(CNC(c2cc(C#N)no2)=O)NC(N2CCCC2)=O)cc1 c1(C(=O)NCCC(CC)(CC)NC(CSCC)=O)ccc(F)c2c1CCC2 c1(C(N(CCNC(c2cnnn2C2CC2)=O)CC)=O)cc(C)n(C2CC2)c1C C1(NC(c2ccc(OC(F)F)cn2)=O)CCN(C(c2ccnnc2)=O)CCC1(F)F Cc1cc(CC(N2CCOC(CNC(c3ncnc(C)c3C)=O)C2)=O)cc(C)c1 N1(C(C(CC)(C)C)=O)CC2(C1)CN(C(c1cnc(O)c(C)c1)=O)CCO2 Cc1cc(C(N2CCC(C)(CNC(C34CC(O)C3C4)=O)CC2)=O)c(N)cc1F c1(C(=O)NCCC2(O)CCN(C(C(C)OCCC=C)=O)C2)cc(F)cc(Cl)c1 C1(C(=O)NC2C(C)N(C(c3ccnc(S)c3)=O)CCC2)CC2(CO1)CC(F)(F)C2 CCS(=O)(=O)c1cccc(C(=O)NCC=CCNC(=O)C2=CCCOC2)c1 c1(NC(=O)Nc2cc(C(F)(F)F)no2)cccc(OCCCN2CCOCC2)c1 c1(C(C(=O)NCCN(CCOC)C(c2nc(C(F)F)cs2)=O)OC)cnn(C)c1 C(CCC(=O)NCCCCNC(C1(CCO)CC1)=O)NC(C)=O C(c1nc2ccccc2o1)=CC(N1CCC(C)C(NC(C23CCC2CC3)=O)C1)=O N1(C(=O)C=CC2CCCCC2)CCOCC(NC(C2(F)CCCCC2)=O)C1 Cc1cc(=NCC2CC(=C3CCC3)C2)[nH]c(N2CC3CCC(F)(F)C3C2)n1 C(=O)(C1=NOC(C)C1)NC(CNC(c1c(CC)ncs1)=O)(C)CC N1(C(C=C(C)C)=O)CCC(NC(=O)CCc2n[nH]c3c2CCCC3)C(F)(F)CC1 N1(C(C(C)OCC2CC2)=O)CCC(N(C(=O)C=Cc2cnc[nH]2)CCO)CC1 C12(NC(C3OCCN(C(C(C=C)O)=O)CC3)=O)CC3CC(CC1C3)C2 c1(C(N2CC(C(C(=O)NCCCC(C)(C)O)O)C2)=O)cc(F)ccc1O CN1CCC(C(=O)NCc2n[nH]cc2C(N2CCC(N3CC(O)C3)C2)=O)CC1 C(CNC(c1c(C)nn(CCO)c1C)=O)(C(C)C(C)C)NC(CCOC)=O CCC(C)(C)CC(=O)N1CCOC(CCCNC(=O)CC2COCC(C)(C)O2)C1 C(C(=O)NOCCC1CCCCC1)(C1CCCO1)NC(c1c(OC)nsc1)=O C(C(C)(O)CC(=O)NC12CC(C1)N(C(=O)C=Cc1cnn(C)c1)C2)OC C(=O)(C1CCCc2cncn21)N(CCC)CCNC(C1(C(F)(F)F)CC(O)C1)=O c1(CC(N2C(C)(CNC(=O)CC(F)(F)Cl)CCC2)=O)nc(F)c(F)cc1F C(N=c1[nH]c(=NCCc2csc(COC)n2)c2ncccc2[nH]1)c1ccn(CC)n1 N1(C(C2(C(=O)NC)CC2)=O)CCC2(CC1)CCN(C(c1ccnc(C)c1C)=O)C2 c1(C(=O)NC(CC=C)CNC(=O)C(CCC)OCC)cccc(S(C)(=O)=O)c1 c1(C(=O)OC)cccnc1N1CCN(C(=O)C(C)n2cncn2)CC1 Cc1ocnc1C1CC1NC(=O)C(=O)NC12CC(C(=O)O)(C1)C2 C1(C(=O)NC2C(CCC)C2)(NC(=O)CC2CCOC2)CC(O)C1 CN1CCN(C)C(C(=O)NC2CCCC(C(=O)NCCc3ccccn3)CC2)C1 c1(C(=O)NCC(CCCC)NC(c2cc(C)nc(O)c2)=O)cc(Cl)nc(Cl)c1 c1(C(=O)NCCCCNC(c2c(C(C)C)occ2)=O)ccc([N+](=O)[O-])o1 c1(C(=O)NC2(CNC(=O)C(O)CF)CCC2)c[nH]c2ccc(Br)cc2c1=O c1(C(=O)NC(C)C(C)NC(C2(C#N)CC3(CC3)C2)=O)ccc(S(N)(=O)=O)cc1 N1(C(c2c(C)ccc(OC)n2)=O)CCC2CN(C(C3(N(C)C)CC3)=O)CCC2C1 C1(CCC(=O)NCC2CCN2C(=O)CC2CC(=O)C2)(N(C)C)CCCCC1 c1(CC(N2C3CN(C(CSC(C)(C)C)=O)C(C3)C2)=O)nc(F)c(F)cc1F c1(CCC(=O)NC23CN(C(CC=C)=O)C(C2)C3)cc(OC)ccc1OCC N#Cc1ccc(-c2cc(C(N3CC(CC#N)C3)=O)n[nH]2)cc1F C1(C2CCC2)(CNC(C(C)N(CC)CC)=O)CCN(C(=O)CO)CC1 C(C(F)(F)CCC(=O)NC1C2CCCC12)n1cc(C2C(=O)NCCC2)nn1 N1(C(CCN(C(=O)CNc2cccnc2)CC=C)=O)CCC(OC)C(C)(C)C1 C1(NC(CC(=O)N(C)C)=O)C2CC(O)C1N(C(=O)C=Cc1ccoc1)C2 c1(C(N2CCCC(NC(c3c(C)scc3)=O)CC2)=O)ncnc2c1cnn2C C(=O)(C(F)(F)C(F)F)N1CC(OCC)(CNC(C23CCCC2C3(F)F)=O)C1 Cc1nccnc1C(=O)N(C)CC=CC(=O)NCC1(F)CCN(C)C1 C12(CNC(C3CCCOC3C)=O)CC(OC)(CN1C(c1cc(OC)ccn1)=O)C2 C(=O)(C(C)CN(C(=O)CCc1cn(C)nn1)C)NCC(C)OCC#C C1(CN(C(c2ncc(OC)cn2)=O)CC)CCCCN1C(c1nc(O)c(C)s1)=O c1(C(=O)NC(C2CC2C(=O)O)=O)cc2c(O)c(c1)CN2.N1(CC)C(=O)CSC1=S c1(C(C(=O)NCC2CCN2C(c2nnc(N)s2)=O)OCC)ccc(O)cc1.CC CCC(C(=O)NC1(CO)CN(C(C2(C#N)CC3CC3C2)=O)C1)C(F)(F)F c1(C(=O)NC2C=CCN(C(Cc3ccc(C)o3)=O)C2)ccc([N+](=O)[O-])cc1F C1(NC(C2CN(C)CC(C)O2)=O)CCCC12CN(C(=O)CCc1cncs1)C2 C1(O)(CNC(=O)OCC(c2cccc(C)c2)=O)CCCN(C(=O)CCC2CC2)C1 C(CCC(=C)C)(C(=O)NC1CCN(C2CCCC2)C1)N(CC=C)Cc1ccccn1 CCC(C)C(O)C(C)C(=O)NCC1(F)CCN(C(c2cc(C)cc(C)n2)=O)C1 CCS(=O)c1ccccc1C(=O)NCCC(C)NC(=O)Cc1cncnc1O N1(C(c2c(C)nn(-c3cnn(C)c3)n2)=O)CCN(C(C2CC2C)=O)C(CF)C1 Cc1ccc(=N)[nH]c1C(=O)NC1(CNC(C2CC2C(F)F)=O)CCOC1 N1(C(C2CC(C)C2)=O)CCN(C)C(C(N2C3CSCC2C3)=O)C1 c1(C(=O)NCC=CCNC(C(c2ccc(C)s2)C)=O)ccc(S(N)(=O)=O)nc1 C(=O)(CC(O)CSC1CC1)N(C(C)CNC(=O)OC(C)(C)C)CC C1(CCC)(NC(c2csc(C(F)(F)F)c2)=O)CCCN(C(C2(C(N)=O)CC2)=O)C1 c1(C(=O)NC2CC(CNC(C3C(OCC)C3)=O)C2)csc(-c2ccccn2)n1 c1(CCC(=O)NCC2CCN(C(c3nccc(C)n3)=O)C2)n[nH]c2ccccc12 C1(CNC(C(C)(C)C2CC2)=O)CC2CCC(C1)N2C(c1cnnn1C1CC1)=O C(C(C)CC(=O)NC(C)CNC(c1occ(C)c1C)=O)OC c1(C(C)C)cc(=NC(C)CC(C)NC(C2CCC(C)(C)O2)=O)[nH]c(Cl)n1 C(=O)(C1=CCS(=O)(=O)C1)NCCCCC(C)NC(=O)Cn1nccn1 C1(SC)CCN(C(c2sccc2CNC(C2CCC2C)=O)=O)CC1 c1(CC)nc(C)c(C(N2CSCC2C(=O)NOC2CCCC3CC23)=O)o1 c1(C(N(CC(C)NC(c2n(CC)ncc2)=O)C2CC2)=O)cc(C)c(O)c(C)c1 CC1CN(C(c2ccc(Cc3ccccc3)[nH]2)=O)CC1NC(=O)CCOC1CC1 C1(CNC(=O)CSC(F)F)CCCC2(CN(C(C34CCCN(CCC3)C4)=O)C2)O1 N1(C(c2ccc(NC(C)=O)s2)=O)CCC(C)C(CNC(=O)C(C)=C2CCC2)C1 N1(C(c2c(-c3n(C)ncc3)n[nH]c2)=O)CCCOC(CNC(C2CC2C#N)=O)C1 CC1=CCC(NC(c2ccnc(-c3ccco3)c2)c2nnnn2C2COC2)CC1 c1(-n2c(C)cnn2)ccc(C(=O)NCCNC(C2COCCO2)=O)cc1 C(CC(C(=O)NC(C1CC1N(C)C)=O)NC(c1ccc(C)s1)=O)OC C1(CNC(C(C(C)C)O)=O)COCCN(C(c2nnc(O)cc2O)=O)C1 C12(CC(O)C1)C(=O)N2.C12(C(=O)NC3(COCC)CC3)CSCC1C2 N1(C(C(C(C)C(=O)NC(C)(C)C)(C)C)=O)CCOCC2(CC2)C1 CCC(C(C)C)C(C(=O)NCCOC)N(C)CC1CCS(=O)(=O)C1 C(=O)(C1=NOC(C)(C)C1)NC1C2CN(C(C(N3CCCCCC3=O)C)=O)CC1C2 N1(CCn2c(C)ncc2)CCn2cc(C(=O)NCc3ccc(O)cc3)nc2C1 OC1(C2CC2)CCCN(Cc2cc(I)cc(F)c2F)C1 S(=O)(=O)(c1ccnc(O)c1)N(C(c1c(C)cccn1)C)C c1(CNC(=O)NC(C2CCC(=O)C2)C)cc2ccccc2nc1Cl c1(C(N2CC(CC)(NC(c3cnc(C(C)O)s3)=O)C2)=O)cc(C)n(C(C)C)n1 c1(C(=O)NC2(C)CN(C(C3CCCO3)=O)C2)nc(Br)c2ccccn12 C1(CN(C(C(c2cnn(C)c2)OC)=O)C)CCN(C(C2CCN(C)C2=O)=O)CC1 N#Cc1ccc(CC2CCCCN2C(c2ccc(C(F)C(F)(F)F)cn2)=O)cc1 C(C)(C(C(C)C)NC(c1cc(C(C)=O)c(C)o1)=O)NC(c1cn(CC=C)nc1)=O C(CC(C)(C)C)(C(=O)NCC1CN(C(c2csc(CO)n2)=O)CC12CCC2)OC C#Cc1ccc(C(=O)NCC(C2CCOC2)NC(=O)Cc2nnc(S)n2C)cc1 N1(C(CSCC)=O)CCCC(C)(CNC(c2ncc(C)cc2OC)=O)C1 CCCCCC(C(=O)NCC1COCCN(C(c2cc(C)on2)=O)C1)C(C)C Nc1c(F)cc(F)c(F)c1C(N1CC(NC(=O)CCc2cncs2)CC(O)C1)=O C1(C(=O)NC(CCOCCOC)=O)CCN(C(=O)Cc2cc[nH]c2)CC1O c1(C(=O)NCC2N(c3nccc(OC(C)C)n3)CCC2C)c(F)cccc1F c1(NC(N(C2CS(=O)(=O)CC2O)C)=O)cc(Br)cc2c1OCO2 C12(C(=O)NC(CN(C(c3c(CC)nns3)=O)C)C)CCC(C)(CC1)OC2 C(=O)(C1OC(=O)c2ccccc21)NCCCOCCNC(CS(C)(=O)=O)=O N1(C(C(CC(F)F)NC(Cc2n(C)ncc2)=O)=O)CCc2sccc2C1 c1(C(=O)NCC2C(C)CN(C(C3CC(F)C3)=O)C2)ccc(N)c2ncccc12 c1(OC)cc(C(=O)NC2C3CC(NC(C4(CF)CC4)=O)CC23)cnc1O C#CCC(C)(C(=O)NC1CCN(C(C)=O)C1)NC(c1c[nH]c(=NC)s1)=O c1(NC(=O)C(=O)NCCCCN2CCCC2=O)cc(Br)ccc1Cl C1(C)(NC(=O)NC2C(OCC)COCC2)CC(=O)N(C)C1 N1(C(C=C(CC)C)=O)CCC(NC(c2cc(COC)cn2C)=O)C(C(C)C)C1 c1(C(C(=O)NC(c2ccccc2)C)N(CC(C)C(C)C)C)ccn(CCF)n1 N1(C(C(c2ccccc2)OC)=O)CC2(CC(NC(=O)CCn3ccnn3)CO2)C1 C(C(=O)Nn1cccn1)C1(N(C)C)CN(C(c2[nH]cc(C(C)(C)C)c2)=O)C1 N1(C(C2CC(C)(F)C2)=O)CC2CCCC(NC(=O)Cc3cccs3)C2C1 C1(NC(c2c[nH]c(Br)c2)=O)CCCN(C(C2CC(O)CN2)=O)C1 C12(NC3CC3)CCC(N=[N+]=[N-])C1C2.C12(CCC1)CC(=O)N2CC c1(OC)ccc(C(=O)NCC2(CNC(=O)CC3(CO)CC3)CCOCC2)cc1 C1(CNC(c2nc(C(C)C)sc2)=O)CCN(C(=O)CC2CSCCO2)C1(C)C c1(NCC2CCN(C(C3(F)CCC(C)CC3)=O)C2)ncc(C#N)cc1Cl c1(C(=O)N)nc2cccc(F)c2s1.c1(C=O)ccc(C(N)=O)cc1.C12(CC1)CN(C)C2 C1(C)(CNC(C(C2CC2)OCC)=O)CCCN1C(=O)C(=O)C=Cc1cccs1 C(=O)(CCCCC(C)CC)NCC(C(NOCC(CC)C)=O)OC c1(N(C)CC2CCN(C(=O)C(F)n3cccn3)C2)nccc(S(C)(=O)=O)n1 C(=O)(C1CCc2nccn21)N1CC(NC(C(CC)=CCCC)=O)C2C1CCC2 CCCC(C(=O)OC)C(=O)NC(CNC(c1ccc(C(C)C)o1)=O)C1CC1 C1(NC(c2ccnc(-c3cc(F)ccc3CO)c2)=O)CC2(C1)CS(=O)(=O)C2 C12(CNC(C=CC)=O)CC(C(N)=O)(C1)C1(CN(C(C34CCCCC3C4)=O)C1)O2 N1(Cc2ccc(OC(C)C)nc2)CCCCC(NC(C2C3CCCC23)=O)C1 c1(OCC)cccc(C(N2CCCC(NC(C3COCCO3)=O)C2C)=O)c1N N1(C(C2CCCCS2)=O)CC(CNC(C2(c3cc[nH]n3)CC2)=O)CC12CCC2 c1(C(N2C(CNC(c3c(OC)cccc3)=O)CCC2)=O)cc(C)c2[nH]cnc2c1 C1(NC(C(C)(C)Oc2ccccc2Cl)=O)CC2CC1N(C(=O)Cc1ccsc1)C2 c1(OC)ccc(C(=O)NCC2CCCC(NC(=O)C=C3CCC3)C2)cc1OC CCC(CC(F)F)C(=O)NC12CCCN(C(c3cc(C(F)F)nn3C)=O)CC1C2 C(CN=c1cc(C)nc(C(C)C)[nH]1)(C1CC1)NC(C=C(C)C(F)F)=O CC1=CCN(C(C2CC3CC3N2C(=O)C(C)N=[N+]=[N-])=O)CC1 CC(C)C(F)(F)CC(=O)NC1CC(CNC(=O)CCCN2C(=O)CCC2=O)C1 C1(NC(c2n(CC=C)nnn2)c2ccn(CCC)n2)CCCC(C2CC2)C1 c1(C(=O)NC2C(C)(C)N(C(c3ccncc3F)=O)CC2)ccc2ncnn2c1 CCC(CC)(CO)C(=O)NCC1CCCN(C(=O)COC2CN(C(C)=O)C2)C1 C1(CC)CCCC1(C)NC(=O)COC(C)(C)CNC(=O)CN1CCCCC1C N1(C(C(C(C)C)O)=O)CCCC(O)(CNC(c2[nH]ccc2C2CC2)=O)CC1 N1(C(c2ncc(CC)s2)=O)CCN(C(c2cc(Cl)nn2C)=O)CC1C(C)C N1(C(Cc2c(C)occ2)=O)CCN(C(=O)CC2CCCNC(=O)C2)C(CCO)C1 Cc1cc(F)c(-c2nc(Cc3cc(C(C)(C)C)no3)nn2C2CCCC2(C)C)nn1 c1(NCCC(COC)O)ccc(S(=O)(=O)NCCN(CC(F)(F)F)CC)cc1F CN1CCC2CN(C(C3CCCC3NC(C3C=CC(=O)N=N3)=O)=O)CCC12 C(N=c1[nH]c(=N)[nH]c(=NC2CCOC2C(C)C)[nH]1)c1nc(COC)sc1 CCCCCCC(F)C(=O)NC(C)(C)CN(C)C(C1(C)CCN(C)C1=O)=O C(=O)(C1=C(SC)CCCC1)NC(CN(C(=O)Cc1scnc1C)CC)C c1(C2C(C(=O)NC(C3(C(N4CC(n5cnnc5)C4)=O)CC3)C)C2)ccccc1 C1(C(=O)NC(C)(C)CNC(c2cn(CCF)nn2)=O)CCCC(F)C1 C1(CC(=O)NCC(COCCCOC)O)CCCN1C(=O)OC CCCC(CC(C)C)C(=O)NC1CCC(CNC(=O)CN(C)C2CC2)CC1 c1(C(N2C(C)CC(CC(=O)N(CC=C)CCOC)C2)=O)ccn2ccccc12 c1(NCCCCCC)[nH]c(=NCC(C)CC(C)C)nc2c1ncn2C c1(C(=O)NC(C2CC2c2ccc(Br)s2)C)cnc(Cl)c(Br)c1 C1(C(N2CC(C)(CC(=O)Nc3ccc(F)cc3C#N)C2)=O)CCc2nc[nH]c2C1 c1(C(N2C(CNC(C(c3n(C)ncc3)O)=O)COCC2)=O)cn2c(n1)CCC2 Cc1cc(C(=O)NCCC(C)NC(c2ccc(OCCO)cc2)=O)ncc1C#N Cc1c(C(=O)NCC2(CN(C)C(c3c[nH]nc3-c3ccsc3)=O)CC2)ccn1C c1(N(C(=O)CCN(C(C)C)C2CC2)CCC)ncccn1 N1(C(CCCSC)=O)CC(CNC(c2cc(C(N)=O)cn2C)=O)CC(C)C1 c1(NCC(C2CCCCC2)NC(CCC=CC)=O)cccc(NS(N)(=O)=O)c1 N1(C(C2OC3CCC2C3)=O)CCC(N2CCNCC2)CC1 C(CCC(C)C(=O)N1CCC(N(C)C(c2ccc(OC)cc2OC)=O)C1)OC Cc1nn(CC(N2CC3CC2C3CNC(=O)COC2CCC2)=O)c(C)c1[N+](=O)[O-] CCC(C)CC(=O)N1CC(N(C(=O)C(C)=C(C)C)C)C(O)C1 c1(C(=O)NCC(CNC(=O)CC2COC(=O)C2)OC)cccc(F)c1C#N C=C(C)CCCC(=O)NC(Cn1cncn1)C(=O)NCC1C2CCCC12 C#Cc1cn(C)nc1C(=O)NCc1csc(C(=O)NC2(C3CCCO3)CC2)c1 C1(NC(=O)Cc2csc(-c3ccco3)n2)CC2CN(C(=O)C(F)C3CC3)CC2C1 C(C(O)CCNC(C1CS(=O)(=O)C1)=O)NC(COCC=C)=O C(C(=O)N1CCC(C(=O)NCc2cccnc2Cl)O1)C1C(C(C)C)C1 c1(CNC(NCC2C(=C)C2)=NC)cccc(OCCOC)c1 c1(C(=O)NCC2CCN(C(c3cn(CCCC)nc3C)=O)C2)ccc(F)cc1O c1(C(N2C(CNC(C3(C)CC3)=O)CC3CC32)=O)cc2cccn2cn1 N1(C(C=CCC)=O)CCC2CN(C(=O)C(C)(C)C3CCOCC3)CCC2C1 C1(C(=O)NC(C2(CNC(c3c(Cl)nn(C)c3Cl)=O)CC2)C)CC(S(C)(=O)=O)C1 C1(NC(C2(OC)CCOC2)=O)CCC(N(C(=O)CSC2CCS(=O)(=O)C2)C)CC1 N1(C(C(=O)NCC)=O)CC(NC(c2occc2C)=O)CC1(C)C c1(C(N2CC3CN(C(c4n(CC)nc(C)c4)=O)C3C2)=O)n[nH]c2c1CCC2C C1(CNC(C2N(C)CCC2)=O)CCC2(CCN(C(C3COC(=O)N3)=O)CC2)CO1 C1(CC(=O)N(C)CCNC(=O)C=C(C2CC2)C2CC2)Cc2ccc(Cl)cc2C1=O C(N=c1[nH]c(=NC2CC=CC2)[nH]c2c1SCC2)C1(Br)CC1 CC(CCC(=O)NCC1(C#N)CCC1)NC(C1CCSCC1)=O C1(C)(C(=O)NCC(C)NC(c2ccnc(NC3CCC3)c2)=O)CC2CCC2C1 CC(C)(C)CCC(=O)N1CCC(NC(=O)CNS(N)(=O)=O)CC1C1CC1 c1(CSC)ccc(Cl)c(C(=O)NCC2CCCN2C(c2cccc(Cl)c2)=O)c1 C(C)(C(=O)NCC1CCC(NC(=O)CC2CCCO2)C1)(c1ccccc1)N(C)C N1(CC)CCOCC1C(=O)N(CCCCCNC(C1CCCN1CC)=O)C C1(NC(CCCC#C)=O)CC2CC1CC2C(N1CC(=O)NC(C(C)C)C1)=O c1(NC(c2cc(OC)no2)=O)cccc(-c2cnc(CN(C)C)nc2)c1 N1(C(c2c(CC)scn2)=O)CCCC(NC(=O)C=Cc2ccnn2CC)C1C CCC(C)CCC(=O)NCc1cc(O)ccc1C C(=O)(C(C(C)(C)C)N1CCCC1)NCCC1CC(NC(c2c(OC)n[nH]c2)=O)C1 C=Cc1cc(C(N2CC(C)CCC2CNC(c2cnsn2)=O)=O)cc(F)c1 C1(CC(N2CCC(N(CCC)C(c3n[nH]cc3Br)=O)C2)=O)C(C)(C)C1(C)C C(CCCC(CO)NC(c1ccc(C)cc1)=O)NC(c1c(CC)ncs1)=O N1(C(c2cn(C)nc2C2CCCO2)=O)CC2(C1)CN(C(C1(C3CCCO3)CC1)=O)C2 CC1CC2(CC(C(N3CC4C(N(C(=O)Cn5cccn5)C)C4C3)=O)C2)C1 C1(CNC(c2ncn(C)n2)=O)CC12CCN(C(=O)Cc1cc(F)ccc1F)CC2 c1(C2C(NC(C3CC3C(=O)NCCCOCC)=O)C2)c(C)noc1C.COC CN1CCC2CN(C(c3ccc(C(=O)N=S(C)(C)=O)cc3)=O)CC12 C1(C(C)NC(c2c(C)[nH]cc2)=O)CCCN(C(=O)CCCN2C(=O)CNC2=O)C1 C(=O)(C(C(C)(C)C)SC1CCC1)N(CC(C)C)CCO.C1(=O)CN(C)N1 Cc1cn2c(C)c(C(=O)NCC3(C)CN(C(=O)C(CO)N(C)C)CCO3)nc2s1 c1(COCc2onc(-c3c(N)n(C4CC4)nc3)n2)ccc2c(c1)OCO2 N1(C(C(C(C)C)F)=O)CCOCC(CNC(c2ccnn2-c2ccncc2)=O)C1 C1(CNC(C(C)C)=O)CC2(CO1)CN(C(=O)CC1Cn3ccnc3NC1=O)C2 CC(Cc1cnc[nH]1)C(=O)NCC=CCNC(=O)CCCc1nc[nH]n1 Cc1ccoc1CNC(=O)C(c1cnn(C)c1)NC(C1CC1C(C)C)=O CCCC(CC)C(=O)N1CCN(C(=O)C=Cc2ccsc2)C(CC(C)C)C1 C1(C(=O)N)CCCCCC1.C1(C(N(C(C)C)CCN(C)C)=O)CC(C(=O)OC)C1 CCCC(CCC)C(=O)NCC(=O)NCC(=O)NC1(C(=O)NC)CC1 c1(C(=O)NCC(CN(C(=O)COCc2nc[nH]n2)C)(C)C)cc(C#N)ccc1O C(C)(C)(CCn1cccc1)NC(CC1N(C(CSC)=O)CC1)=O N1(C(Cn2c(=O)sc(C)c2C)=O)CC(CO)C2(C1)CN(C(C1CCS1(=O)=O)=O)C2 CC(CNC(c1nonc1N)=O)CC(=O)N(C1CCN(C)C1=O)C c1(C(N2C(CNC(c3ccc(Cl)o3)=O)COCC2)=O)cn2ccsc2n1 C1(CCC)CCCN(C(C2CC(N(C(=O)COC(C)CC)C)C2)=O)CC1 CN1CCC(=CC(N2CC(O)CC2CNC(c2cnc(C3CC3)s2)=O)=O)CC1 N1(C(C(CC)C(=O)OC)=O)CCCC2(C1)CN(C(=O)C(=Cc1ccncc1)C)C2 c1(CC(=O)NC2CN(S(Cc3cccc(N(C)C)c3)(=O)=O)C2)ccc(C#N)cc1 N1(C(COCCCC)=O)CCC2(CCC(CNC(C3CC3(F)F)=O)OC2)CC1 c1(CC)cc(C(=O)NC2COCC2NC(c2ncnn2CC)=O)nn1CCO c1(NCC2OCC(C(=O)O)C2)cc(Br)c2c(c1)OCCO2 C1(c2ccc(C)o2)CCCCN1CC(c1ccc(C(F)(F)F)cc1)N CCCCC(C)CCC(=O)NC(C)(CNC(c1ncc(Cl)cc1Cl)=O)CO c1(CNCC(CO)F)cccc(F)c1I c1(CC(N2C3CCC(C3)C2CNC(=O)C(F)(F)CO)=O)cccc2nsnc12 N1(C(c2cc3nc(C)sc3[nH]2)=O)CCN(C(C2(C)CCCN2C)=O)CC12CCC2 CCC(C(=O)N1CC(C(C)NC(C2(CC)CC2(F)F)=O)C1)N(C)C c1(C(=O)NC2(CNC(CC)=O)CC2)ccc(Sc2ccncc2)cc1C N1(C(CC2(NC(CC3C(CC)C3)=O)CCC2)=O)CCCC(C)(CC)C1 Cc1ccc(C(=O)NC2CCCC(NC(C3(C)CC4CC4C3)=O)C2)cc1Cl C1(C(=O)NCc2cccc(CNC(=O)C=CBr)c2)CCS(=O)(=O)CC1 N1(C(C2CCCCS2)=O)CC2CC(C1)N(C(c1ccnn3ccnc13)=O)C2 CC1CCC(C(N2CC(C3CCCCO3)C2)=O)N1C(c1cnc(O)[nH]1)=O C1(NC(C2(C)CC2(Cl)Cl)=O)CCCCN(C(=O)CCOCC(F)F)C1 C1(C(=O)N(C)Cc2cn(C(c3ccccc3Cl)C)nn2)(CC)CCCC1O C1(C(N(C2CCCC2)CCCC)=O)CN(C(=O)C=CCCC)CC12CC2 N1(C(CCC=C)=O)CC(C(=O)Nc2ccc(OC)cc2C)N2CCC1C2 C=CC(CCC)CC(=O)N(C)CCN(C)C(c1c(C)ncc(C)c1O)=O CC1CC(=O)NCCN1CCC(C(=O)NCC(F)(F)F)C1CCC1 C(=O)(CCCS(N)(=O)=O)N(c1n[nH]cc1[N+](=O)[O-])C1CC(C)N(CCCCCC)C1 N1(C(CSCC)=O)CCN(C(c2ccc(N)c(SC)c2)=O)CC1CF CC(C)C(CCN(C)C(C1(CCF)CC1)=O)NC(c1nncn1C)=O N1(C(CCCC=C)=O)CC(C(=O)NCC(=O)NC(C)(C)C)CC(C)C1 C=CC1(C(=O)Nc2cccnc2)CCN(C(=O)C(=Cc2ccccc2)C)C1 c1(CC(=O)NC2(CNC(C3CC4C=CC3C4)=O)CC2)c(F)cccc1F C1(CCNC(CCN(S(C)(=O)=O)C)=O)CCCN(C(C2(C)CC=CC2)=O)C1 c1(NC(C23CC2CN(c2ccnc4ccnn24)C3)=O)cc(O)ccc1[N+](=O)[O-] CCCC(CNC(=O)CC(C)c1ccco1)C(=O)NC(c1ccc(O)cc1)C c1(C(=O)NCCCN(C(c2c(C(C)C)c[nH]n2)=O)C)c[nH]c2cnccc12 CC1(C)C(CNC(C2CCS(=O)(=O)N2)=O)CCN1C(c1nccc(Cl)c1O)=O c1(CC)ccnc(C(N2CC(OC)C(NC(c3n[nH]cc3OC)=O)C2)=O)c1 c1(C(=O)NCCC2CCCN(C(CCCCC=C)=O)C2)nn(C)c2c1CCC2 c1(C(C)CC(=O)N(C(C)CCNC(c2cncs2)=O)C)ccccc1F c1(C(N2CCC(C)(C(=O)Nc3ccc(O)c(F)c3F)C2)=O)cc2cnccc2[nH]1 Cc1oc(C(C)(C)C)cc1C(=O)NCCCNC(=O)Cc1cc(Cl)sc1Cl CN1CCCC(CC(=O)NC2CCCC2C(=O)N(CCO)CCN2CCCCC2)C1 N1(C(C2N(CC)CC2)=O)CCCC2CN(C(C3CC4CCC3CC4)=O)CC12 CC(CC(F)F)C(=O)N(C(C(N1CCC(F)(CO)C1)=O)C1CC1)C C(=O)(C(C)(C)NC(=O)Cc1ccccc1)NCC(CN(C(C(F)=CC)=O)C)C CC1C(NC(=O)Cc2cn[nH]c2)CCCN1C(=O)CCC(=O)c1ccc(F)cc1 CCC(F)(C(=O)OC)C(=O)N1CC(CCNC(c2cc(C(F)(F)F)nn2C)=O)C1 C(CCN=C(NC(c1cccc(C(F)(F)F)c1)C)NC1CCC(C)(C)C1)OCC CN1CCCC(N=c2[nH]c(=N)[nH]c(=NCC3CC3C3CCOCC3)[nH]2)CC1 N1(C(Cc2c(C)n[nH]c2C)=O)C2CCC1CN(C(C1(C(C)C)CCCC1O)=O)C2 c1(C(N2CC(NC(C(CSC)C)=O)C(CC3CCCC3)C2)=O)ccc(F)cc1F N1(C(C2CCCN(C(=O)OC)C2)=O)CCCC12CCCN(C(c1cnc[nH]1)=O)C2 c1(C(N(C2CCN(C(C3CC(C)C3)=O)C2)CCO)=O)cc(C#N)ccc1O CC1(C)COc2cc(C(=O)NCc3csc(Br)n3)nn2C1 O=C(C1=CC2(CCN(C(=O)C(O)Cn3cncn3)C2)C1)NCc1ccc(O)cc1 N1(C(c2cnc(C(C)OC)s2)=O)CC(NC(c2cc(C)cnc2N)=O)CCC1C N1(C(CC(C)OC)=O)C2COCC1CC(NC(=O)CN(C)Cc1ccccc1)C2 C(=O)(CC(C)c1cnn(C)c1)NC(CC)CN(C(C1CC(OC)C1)=O)CC c1(C(=O)OCC)sc(Cl)c(Cl)c1Nc1ccc(O)cc1 C1(C(=O)NC(CCNC)c2cccs2)CCC(=O)NC1.n1(CC(=O)N)cncn1 c1(OC)ccnc(CNC(=O)CCC2CCCN2C(C2C(C)C2C)=O)c1 c1(C(=O)NCC2CCN(C(C3C(C)(C)COCC3)=O)C2)cnc2[nH]ccnc1-2 CCC(C)(CCC(C)C)C(=O)NC12CCCC1N(C(=O)C(C)NC(C)=O)CC2 c1(C(=O)NC2CN(C(C(CC#C)O)=O)CC(C)(C)C2)cnc(O)c2ccccc12 Cc1oc(CNC(C2CC3CCC2O3)=O)nc1C(=O)NCCc1cn(C)cn1 C(C(C)(C)C(C)(C)O)NC(C1CCCN(C(c2nc(CC)oc2C)=O)C1)=O c1(C(=O)NCC2CCC(C)N(C(c3cc(C)n(C)n3)=O)C2)cc(F)c(F)cc1O c1(NC(C2C(CNC(C(c3ccccc3)C)=O)C2)=O)cnc(Cl)nc1 c1(C(=O)NCCC(C)NC)ccc(Cn2ccnc2C)cc1 C1(CC(N2CC(O)(COC)C2)=O)CN(C(c2cc(OC)cs2)=O)CCC1C C1(C(=O)NCC2(NC(CN(C)C(=O)C3CC3)=O)CC2)Cc2cc(Br)ccc2O1 CC(C)(F)CCC(=O)NCC1(C)CN(C(c2cnc(C(F)(F)F)s2)=O)CCO1 c1(C(N2CCC(NC(C(C(C)C)C)=O)C23CCC3)=O)ccc2ncncc2c1 N1(C(CCCCC)=O)CCN(C)C(C(N2C(CO)CCC2CO)=O)C1 c1(SC)cc(C(N2CC(CNC(c3ccc(O)cn3)=O)C2)=O)ccc1F C1(NC(C2CCC(CC)O2)=O)CN(CC)C(C)(CC)C1.c1(C=O)cc(Cl)c(C)cn1 C(CCN=c1c(C#N)c[nH]c2c(F)cc(F)cc12)NC(C1C(C)(C)S(=O)(=O)CC1)=O CC1(C)C(NC(=O)C(=O)NC2CCCCC2)CCN1C(=O)CCNC(=O)CO N1(C(C=COCC)=O)CC2CCN(C(C3CN4CCCC4CO3)=O)C2C1 N1(C(Cn2c(C(C)C)ncc2)=O)CCC(C)C(CNC(C23CC(C)(C2)C3)=O)C1 C1(C)(C(=O)NCC(C)(C2CCC2)NC(=O)C(C)(C)n2cccn2)C=CCC1 c1(C(=O)NC(CC)CNC(c2c[nH]c(C)c2)=O)cn(C)c(=O)nc1O CC(C)CC(C(=O)NCc1cccc(O)c1)NC(c1ccc(C2CC2)cc1F)=O C1(NC(CCC=C)=O)CN(C(c2cc(N)c(O)c(F)c2)=O)C2(CCOCC2)C1 C1(CNC(Cc2c(C)ncs2)=O)CC(C(F)(F)F)CCN1C(=O)CCS(N)(=O)=O c1(OC)cc(C(N2CCC2CNC(=O)CC2CCCC2)=O)cc(F)n1 C1(N(C(CC2(CC)CC2)=O)C)CCN(C(c2c[nH]nc2OCCC(F)F)=O)CC1 c1(OC)ccc(NC(=O)C=CC(C)NC(C2COC(=O)C2)=O)cc1C C=C(C)CCC(=O)N1CC2C(CNC(c3c[nH]nc3OC)=O)C2C1 S(=O)(=O)(c1cccnc1NC(CC)COC)NCC(O)C1(Cl)CC1 N1(CC2C(C)(C)C(NC(=O)CN(C)C3CC3)C2)CCOC(C)(C2CC2)C1 C12(C(N(CC(CNC(C(CC)(F)F)=O)O)C)=O)CCC(CC1)C2(C)C N1(C(CC(C(=C)C)OCC)=O)CCC2(C1)CN(C(c1c(Cl)cnn1C)=O)CCO2 c1(CC)cccc(F)c1NC(=O)CC1CCCCN1C(=O)COCCF CC(C)=C=CC(=O)NC(C1CCN(C(c2ocnc2C)=O)CC1)C C1(N(C(CCC2C(C)C2)=O)C(C2CC3CCC2CC3)=O)CC2C(O)C(O)CC12 C(=O)(C1CCCc2cccnc21)NC(CNC(=O)CC1(O)CCCCC1)CO C1(NC(c2nccc(N(C)C)c2)=O)CCCN(C(=O)CCNC(=O)CO)CC1 c1(CCC(N2CC(C)C(NC(c3cc(Cl)cnc3O)=O)C2)=O)cc(F)cnc1O N1(C(C2CCC(CC)O2)=O)CCC(NC(=O)CCn2ccc(C)n2)CC1C C1(CNC(C(C)=C2CCC2)=O)CCCN1C(=O)C(=Cc1cn[nH]c1)C Cc1ccc(F)c(C(=O)NC(C)C(=O)NC(c2cccnc2)CO)n1 CCC(C)(C#N)C(=O)NCC(C1CCC1)NC(c1ccnc(C)c1O)=O N1(C(c2cc(C)ns2)=O)CCCN(C(=O)COCC2CCCOC2)C(C(C)C)C1 C(=O)(CCCC(=O)C(C)(C)C)N1CC(CC)N(C(=O)CN2C(C)CCCC2C)CC1 N1(C(C(c2ccc(C)cc2)=O)=O)CCC2(CCC2)C(NC(=O)CN(C)C(N)=O)C1 c1(C(=O)NCC2(CN(C(=O)CCC3CC3)C)CC2)cnc(-c2ccccc2)o1 C(=O)(C(CNC(C1CCCO1)=O)CC(C)C)NCc1c(CC)onc1C C1(CC(N2CCC(N(C)C(c3cc(C(F)F)no3)=O)C2)=O)CC2(CCC2)CCO1 N1(C(C(c2ccc(F)cc2)OC)=O)CC2CC2(C)C1 C12(NC(Cn3ccc(C)n3)=O)CCOCC1CN(C(c1[nH]c(C)cc1C)=O)C2 C1(CC)COC(C)CN1C(C1CN(C(=O)CCc2cncs2)CC(C)O1)=O N1(C(CC2CC(=C)C2)=O)CC(NC(=O)C(C)(C)F)C(C)C1 NC(=O)CC(C(=O)N1CCCc2ccnn21)NC(=O)Cn1[nH]cnc1=N CC(C)CCC(=O)NC1CCCC1N1CCN(C(c2ccccc2OC)=O)CC1 N1(C(C(CC)COC)=O)CC2CCC(CNc3ncc(F)c(OC)n3)(C2)C1 c1(C(N2CC(C)(C(=O)NC(c3ccsc3)C)C2)=O)ccc2occc2c1 c1(OCC)ccc(C(=O)N(C)CC2CCN(C(C3CCCCN3C)=O)C2)c(F)c1 N(C(=NCCCOC)NCc1ccccc1)CC(=O)NC.C1(C)CCN1 C(C(F)(F)CCC(=O)OC)OCc1cccc(-n2cc(-c3c(C)ccs3)nn2)c1 CC1(C)CC2CN(C(=O)CC3CC4(CC4)CO3)CC12 c1(C(C)CC(N2CCOC(OC(C)(C)C)C2)=O)c[nH]c2ccccc12 N1(C(=O)NC(c2ncc(-c3ccccc3)[nH]2)C(C)C)CC(F)C(F)C1 C(CC(C(C)C)NC(C1CC1c1ccsc1)=O)NC(CC(=C)C)=O S(=O)(=O)(c1ccc(N2CC=C(C(C)(C)C)CC2)c(F)c1)NCc1ncc(C)nc1 C1(C(N2CC(O)(c3cn(-c4ccc(CO)cc4)nn3)C2)=O)C2CCCCCCC12 N1(C(C2(C)CNC(=O)C2)=O)CC2CC(C1)N2C(C1(F)CCCCC1)=O c1(CC(=O)NCC2(OC)CN(C(=O)Cc3ccoc3)C2)ccccc1Br C(C(=O)N=c1cco[nH]1)N1CC(CN(C)C(c2ccnc(F)c2F)=O)C1 C1(C(=O)NC(c2csnn2)C)CN(C(=O)CC(C)(C)C(F)F)CC(C)(C)C1 C1(C)(C(N(CCOCCCN(C(C(CC#C)C2CC2)=O)C)C)=O)CCCN(C)C1 c1(C(=O)OC)cc2c(C)cccn2n1.c1(C(=O)NC2CC(N)C2)cnc(CN)nc1 Cc1cc(C(N2CCC(C)(C)C2CC(=O)NCC2CCN(C)C2)=O)cc(C)c1 C1(C(=O)NC2C3CCN(C(CCC=CC)=O)C32)Cc2ccccc2O1 C(=O)(C(CC(C)(C)C)N(C)CCN1CCCCC1)NC(C)C C1(NC(C2C(C)(C(C)C)C2)=O)CCC2CN(C(=O)Cc3cnn(C)n3)CC2C1 C=CCCCCC(=O)NCC1(NC(c2ccc(O)c(Cl)n2)=O)CCCCC1C Cc1sc(O)nc1C(=O)NCC(CO)NC(=O)CC1CCC(=O)CC1 C1(C(=O)NC(C)CCNC(c2ccnc3ncnn23)=O)Cc2cc(Cl)ccc2O1 C1(C(N2CC(CC=C)(C(=O)NCCc3nncn3C)C2)=O)CCN(C)C1=O Cc1ccc2scc(C(c3nnnn3C(C)(C)C)Nc3cc(C)c(C)s3)c2c1 N1(C(C(N2CC(C)OC(c3ccccc3)C2)=O)=O)CC2CCCN2CC1CO c1(C(N2CC(NC(=O)CC3CC4CC4C3)C(CO)CC2)=O)cc2ccccc2o1 c1(CC(=O)NC(C)C=CC(=O)NCC2(C)CSC2)nocn1 c1(C(=O)NCCCNC(C2(C(=O)OC)CNC(=O)C2)=O)nc(OC)cc(OC)n1 C1(N(C)C)CN(C(C2CCCN2C(=O)CCCn2ccnc2)=O)CC1(C)C C1(CCNC(Cc2cccc(C)c2)=O)CCN(C(c2ccon2)=O)C(C)C1 C1(C(=O)NCC(CN(C)C(C2(CO)CC2(F)F)=O)(C)C)C2CCCCC12 C(=O)(CC(C)CCC(=O)NCCCCCCNC(=O)CC(=O)NC1CC1)OC c1(NC(C(COC(C)C)NC(C(CCCC)F)=O)=O)cnc(C)c(C)c1C c1(C(N2CCN(C(C3CC(CC)C3)=O)CC(O)C2)=O)ncnc2c1ccn2C c1(Nc2cc(C3(C)CC3)ncc2)ccc(S(=O)(=O)N2CC3CC3C2)cc1Cl c1(CC(=O)NCC(CNC(c2c(CC)ocn2)=O)OC)ccc(OC)cc1F N(C(=NCC#Cc1ccccc1)NC1CCC1)C1C(C)(C)CC1 C1(N(C(CN(C(C)=O)C)=O)C)CN(C(=O)N(S(C)(=O)=O)C(C)C)CC1O C(=O)(C(C)(C)CC(=O)NC(CC1CC1)C(=O)NCc1nn[nH]c1C1CC1)OC N1(C(C(=O)NCC)=O)CCCC(C)(C)C1CNC(=O)C=C(C)c1ccccc1F CCC(CC(=O)NC(c1nccc(C)n1)C)N(C(=O)C(c1cccnc1)OC)C C(=O)(C(CCC(N)=O)N(C)C)NCCC1CCN(C(c2ccc(C)cc2C)=O)C1 N1(C(Cc2scc(C)c2)=O)CCC2(CCN(C(c3cccc(C)c3C)=O)CC2)C1 C=CCC(C)(C)CC(=O)N1CC2(CC2)CC1CNC(=O)C(C)n1cccn1 C1(CNC(C=C(C)C(C)C)=O)(NC(=O)C(F)CC2CCC2)CCCC1 CC(C(C)(C)NC(=O)C=Cc1cscn1)NC(c1cc(Cl)no1)=O N1(C(c2n[nH]c(C)c2C)=O)C2CCC1C(CNC(c1ccc(Br)cc1)=O)C2 N1(C(CCCCC)=O)CCOC2(CCN(C(c3cccnc3C)=O)CC2)C1 CCC(CC(=O)N1CC(CC(C)NC(c2cccc(C(C)(C)C)c2)=O)C1)C(F)F c1(OC)ccc(C(=O)NCC2CCN2C(=O)CCCN(C)C(C)=O)c(F)c1 c1(SCC)cc(C(=O)NCC2CCCN2C(=O)C(C)C2CCC2)ccn1 Cc1ccc(CN2CC(NC(C3CCCN(C(=O)C4CC4)C3)=O)C2)c(F)c1F C1(C(=O)NCC(C2CC2)SC)CCCC(NC(=O)C(C)CC#N)C1 C12CC(C1)C(=O)N2C(C)=O.C(CCN)NCC C1(C(N2CC(CNC(C(C)(C)N(C)C)=O)CC2(C)C)=O)CCc2ccnn2C1 c1(C(=O)NC(CNC(C2=CCCCC2C)=O)C2CC2)c[nH]c2cccc(C#N)c12 C1(OC)CC(CNC(=O)Cc2nnc(C)o2)N(C(C2(c3cc[nH]n3)CC2)=O)C1 Cn1ncc(C(=O)NC(CCC2CCC2)C(=O)NCCCN2CCC2)c1N C1(NCC2(c3ccc(Cl)cc3Br)CC2)C2(CCC2)C12CCC2 N#Cc1c(N2CCCC(CNC(C3CCCCO3)=O)CC2)ncc2c1CCC2 C1(NC(C2C(C(=O)OC)C2)=O)CC(OC)CN(C(c2cc(C(N)=O)[nH]n2)=O)C1 Cc1ccc(C(=O)NCC(O)CN(C(=O)CCC2CC3CCC2C3)C)nn1 c1(C(=O)NC(C2CC(NC(Cn3ncc(C#C)c3)=O)C2)C)cccc2nncn12 CCC(C)(C(=O)N1CCC2CN(C(c3coc(C4CCC4)n3)=O)C2C1)C(N)=O C(=O)(C1=NOC(C(N2CC(O)(CNC(C3(CCF)CCOCC3)=O)C2)=O)C1)OC C(=O)(C(O)C(F)(F)F)NC(C1(CNC(c2cnccc2Cl)=O)CC1)C c1(C(=O)NC2CC(NC(C3N(C(C)=O)CCC3)=O)C2)c(C)ccc2ccccc12 C(C)(C(CC(=O)NCC1(OC)CCC(C)C1)NC(=O)CC1CC(N(C)C)C1)OC C(C(C)COCC)NC(C1CC(NC(C2C(CCC)C2)=O)C1)=O C(=O)(CC1=NNC(=O)C1)N1CCN(C(CC2CC(C)C2)=O)CC1CF C(c1cc(C)c(C)cc1C)=Cc1cn(CC=C)nc1 c1(C(=O)NC2C(CNC(CC(C)C3CCCCC3)=O)C2)ccn2nnnc2c1 CCCC(CCC)C(=O)NC1CC1CNC(=O)Cc1cccc([N+](=O)[O-])c1 c1(NC(c2cccc(C(=O)OCC)c2)C)cc2ccc(OC)cc2cn1 Cc1ccc2sc(C(N3CCC(C)(CNC(=O)Cc4cn(C)nn4)C3)=O)cc2c1 c1(OC)ccc(C(=O)NC2(CC3CC3)CCC2)cc1[N+](=O)[O-] c1(C(=O)NCC2(CN(C)C(c3c[nH]nc3F)=O)CC2)cc2ccc(Cl)cc2o1 c1(C(=O)NCC2C(NC(C3(C)CCCO3)=O)C2)ccnc(-c2ccccc2)n1 C1(NC(c2cc(F)c[nH]2)=O)(CO)CCN(Cc2ccc(Cl)cn2)CC1 CC(C)(CC(F)F)C(=O)N1CCCC(O)(CNC(=O)CCC2=CCCC2)C1 CC(C)CC(C)C(=O)N1CC(CNC(=O)COC2CCCC2)C(C(F)(F)F)C1 c1(C(N(C)CC2N(C(c3n(CCC)ncc3)=O)CCC2)=O)c(OC)cccc1F c1(NC(C=CC=CCC)=O)nc(C2CCC2)ncc1F C1(CC)CCCC1(C)C(=O)NC1(C(N2C(C(=O)OCC)CC2C)=O)CC(O)C1.C1(C)CC1 C1(CC)CN(C(c2cc(F)n(C)n2)=O)CCN1C(C1CCC(C)(C)C1)=O CC1CCC(NC(=O)Cc2cnccn2)CN1C(=O)CC1CC2C=CC1CC2 N1(C(COC2CCN(C(C3=CCCC3C)=O)C2)=O)CCn2ncnc2C1 N1(C(c2cn(CC)nc2)=O)CC(NC(=O)CC2CCC(C)O2)C(CC(C)(C)C)C1 C1(CNC(CC2(C=C)CC2)=O)CN(C(c2cc(C#N)c[nH]2)=O)C2(CCC2)C1 Cc1cnn2ccc(C(=O)NC3CC(NC(c4nc(Br)cnc4N)=O)C3)nc12 c1(CC(N2CCN(CCN(C(CCC#C)=O)C)CC2)=O)c[nH]c2cc(F)ccc12 C1(C(=O)NC(C2C(NC(c3cnsn3)=O)C2)=O)COC(Cn2cccn2)C1 Cc1cc(O)n2ncc(C(=O)NC34CCCC3N(C(=O)C(C)CF)CCC4)c2n1 C1(C(=O)NCC(C(C)C)NC(C2CC(n3cnnc3)C2)=O)CCCCC1O Cc1nc(C(N2CC(C3CN(C(c4ccccc4)=O)CCO3)C2)=O)sc1C n1(CCC)cc(C(=O)NC(C2(O)CN(C(=O)Cc3cnn(C4CC4)c3)C2)C)cn1 C(=O)(C(F)C(F)(F)F)NCC(CCCC)NC(C1CC(=O)CC(=O)C1)=O C1(C(CO)NC(CSCC)=O)CCN(C(=O)CCc2nc(C(C)OC)no2)CC1 c1(N)cc2ncccc2[nH]1.c1(N2CCCC(C(C)=O)CC2)cnc(C#N)c(C)n1 C1(C(=O)NCC2CCCN(C(C(CC)C)=O)CC2)CC2(C1)CC1(CC1)C2 N1(C(CC(CC)OC)=O)CCN(C(c2coc(C(C)(C)C)n2)=O)CCC1C C1(CNC(C2(CC=C)CN(C(c3cnsc3C)=O)C2)=O)CCCCC1C c1(C(=O)NC2C(NC(CC3(COC)CCOCC3)=O)C2)cc2cccnc2[nH]1 C1(CNC(CC(=O)N(C)C)=O)CC2CCCC2N1C(c1nnn2c1CSCC2)=O C1(CNC(C2CC3(CN(Cc4c(C)coc4C)C3)C2)=O)=CC2C(=NNC2=O)C=C1 CCCC(CCC)C(=O)N1CCC(F)(C(N2CCC(CC3CC3)C2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)N(C(C)CNC(c1ccc[nH]1)=O)C C(CN=c1nc2sccc2c(N2CCC3C(C)C3C2)[nH]1)CC(N1CCCCC1)C c1(CNC(=O)CC2CC(Cn3cc(Br)cn3)C2)ccc(C(=O)O)cc1F c1(CCC)cccc(C(N2CCC(OCCNC(=O)C=C3CCCC3)C2)=O)c1 C1(C(N2CCC(C(F)(F)F)C2)=O)CCCC(c2nn[nH]n2)C1 c1(CC(=O)NC(C)C=CC(=O)NC2(CN(C)C)CCCCC2)cccc(F)c1O N1(S(C)(=O)=O)CCCc2cc(-c3nc(-c4ccncn4)no3)ccc21 N1(c2ccnc(C(CC)C)n2)CC2CCC(NC(=O)CS(N)(=O)=O)CC2C1 C(=O)(C(=O)N(O)C(C)C)N1CCC(n2cc(CN(S(C)(=O)=O)C)nn2)C1 N1(C(C2CCCC(C)C2)=O)CCCOC(CNC(c2ccnc(F)c2O)=O)C1 CC1(C)CC(C(=O)Nc2ccccc2)CCN1C(=O)CCC(=O)N1CCCC1 c1(CC)cccnc1C(N1CC(CNC(C23CCC2C3)=O)C(O)C1)=O N1(C(C(C)CSN2C(=O)CCC2=O)=O)CC(C)CN(c2ncccn2)CC1C c1(C(=O)NC2C(C(=O)Nc3c(C)c(O)ccc3)C2)c(F)ccc2[nH]ccc12 N1(C(C=CC)=O)CCN(C(c2cnn(C(C)C)c2C)=O)C(CF)C1 Cc1cc(Sc2c(Br)nnn2C)nc(-c2ccc(C)o2)n1 C=CCCN=C(NCCCC1(C)CC1)NCC1CC(=O)N(C)C1=O C1(O)(CNC(c2n(C=C)ncc2)=O)CCN(C(C2(CCCC)CCCC2)=O)CC1 C1(CC(=O)NC2CC2(C)C(C)C)(OC)CN(C(=O)Cn2cncn2)C1 C12(C(=O)NCc3cccc(CC)c3)CCC(CN(C(=O)C=CC3CCCC3)C1)C2 CCCC(C)C(=O)NC(c1ccccc1)CNC(=O)C(N)=O N1(C(CCOCCN(C)C)=O)CCCCCCC1C(=O)NCc1ccnc(O)c1 O=C(C1=CS(=O)(=O)CCC1)NCC1(F)CCCN(C(C23CC(CN2C2CC2)C3)=O)C1 c1(C(N2C(CCNC(=O)COCC3CCC3)CCC2)=O)cnnc(O)c1 c1(CC(=O)OCCn2nc(Br)nc2C2CC2)nnc(C(F)(F)F)s1 c1(N2CCC(F)(CNC(c3ccc(OC)nn3)=O)CC2)nc(C#N)ncc1Cl c1(CN2CCN(C(C3C(CC)OCC3)=O)CC2)cc(OC)c(OC)c(F)c1 C1(C(=O)OCC2CC(COC)C2)CC12CCOc1ccccc12 CCC(CN=c1cc[nH]c(=NCCC)[nH]1)c1ccc(C)c(C)c1 C1(NC(C(C)(C)c2ccsc2)=O)CCN(C(c2ccc(Cl)o2)=O)C12CCC2 C(=O)(C(CC(C)C)n1ccnc1)N1CCC(C(C)NC(CCNC(C)=O)=O)CC1 Cc1nccc2c1CCN(C(c1ccc(F)c(Br)n1)C(=O)NCC(C)C)C2 c1(C(=O)NC(CC(C)NC(c2coc(C(F)F)n2)=O)C)ccc2cccnc2n1 C(=O)(CCC(C)(C)F)N1CCC(C(=O)NCCC2C(C)OCC2)CC1 C1(N(C(C(C)Cc2cccnc2)=O)C)CN(C(=O)C=Cc2ccoc2)CC12CC2 C1(C)(NC(c2cc(SC)on2)=O)CCN(C(C2CCCN2CC)=O)C1.C(C)(C)(C)O N1(C(COC(C)(C)C)=O)CCC(C(=O)NCC2CCNC(=O)C2)C2CCC12 Cc1cnccc1C(=O)NCCCCN(CCCNC(=O)C(C)C1CCOC1)C c1(N(C)Cc2ncc(C)nc2)nc(=NC2CCC(F)CC2)[nH]c2ccccc12 C(=O)(CCCCC(F)(F)F)NCC(C1CCC1)NC(C1N(C=O)CCC1)=O c1(C(=O)NCCN(C(=O)CCn2cnc(=N)[nH]2)C(C)C)noc2c1CC(C)CC2 C1(C(C)C)COCCN(c2nnc(CC(=O)N(C)C)n2CCC(C)(F)F)C1 c1(OC)cc(COC(C2(C)CC(=O)N(C)C2)=O)cc(Cl)n1 C(=O)(C1=NN(C(C)C)C(=O)CC1)N(C1CCN(C(C2C(=C)C2)=O)C1)CCO Cc1nccn1CCC(=O)NC1CC(C)(NC(=O)CC2CCOC2C)C1 c1(CC(N2CCC(NC(C(C(C)C)SCC)=O)C2)=O)c(C)cccc1C C1(NC(C(C)OCC=C)=O)CCN(C(C2CCC(NC(C)=O)CC2)=O)C12CC2 C(=O)(C(C)(C)CF)NCCN(C(=O)C(=O)NCCOC)CC N1(C(c2cn(CC3CC3)nn2)=O)CC23CCCC2(C1)CN(CCCCCC)C3 c1(CC)cc(CC(=O)NC2CC(O)(CNC(=O)COC3CCC3)C2)on1 c1(C(N2C(CNC(C3CC(N(C)C)C3)=O)CCCC2)=O)ccn(CCO)c(=O)c1 C(C)(C(=O)N(CCC(=O)N1CCC1C1CCCC1)CCO)SC.C(CS)NC(C)=O c1(C(C(=O)NCC(C)NC(=O)C(C)c2ccco2)O)ccc(F)c(Cl)c1 CCCCCC(O)CC(=O)NC(C(=O)NCc1ncnn1CCC)C(C)CC c1(C(N2C3CN(C(CCS(=O)(=O)NC)=O)C(CC3)C2)=O)c(C)nc2sc(C)nn12 c1(C(=O)OC)cc(Br)ncc1NCC1CCN(C(c2ccc(Cl)cc2O)=O)C1 c1(C(N(C(C)CNC(=O)Cc2cc(F)ccc2Cl)C)=O)cc(Cl)c(F)cc1F C1(NC(CN2C(C)CC2)=O)CCCCCN(C(c2c(F)cccc2Br)=O)C1 C1(C(=O)NCC(CNC(c2nc(COC(C)(C)C)oc2)=O)F)CCCS(=O)(=O)C1 c1(OC)cc(C(N2CCC(C)(C(=O)O)C2)=O)nc(C(F)(F)F)n1 C1(NC(C=CCCC)=O)CCCCC12CCN(C(=O)C=Cc1cnc(C)s1)CC2 c1(C(=O)NCCC2(NC(CCNC(C)=O)=O)CC2)ccc(S(=O)CC#N)cc1 Cc1ccc(=O)n(CC(N2CCC(NC(c3c(C)cncc3C)=O)C(F)C2)=O)n1 C1(O)(CNC(c2cnc(Cc3ccccc3)s2)=O)CN(C(C2C3CCCC23)=O)C1 C(C)(C)(C(=O)N1OC2CCC1CC2)C1C=CC(NC(C(C)C2CC2)=O)C1 c1(C(N2CCC(NC(C(CC(C)=O)C)=O)C(F)C2)=O)cc(F)cc([N+](=O)[O-])c1Br Cc1cc(CC(=O)NCc2c[nH]nc2C2CCN(C(=O)C(C)C3CC3)C2)n[nH]1 N1(C(c2cc(CC)[nH]n2)=O)CCCC2(NC(c3ccccc3OC)=O)CC12 c1(C(N2CC(N(C(c3nnc(C)s3)=O)C)C2)=O)cc(CC)ccn1.C(C)(C)C C1(N(C(=O)COCCCc2cn(C(C)C(=O)O)nn2)C)CCC(F)(F)CC1 CCCC(C)(O)CC(=O)NC1(CCOC)CCN(C(c2ncc(C)cc2C)=O)C1 c1(OCCOCCO)ncc2c(O)nnc(O)c2n1.C12CC1C(=O)NC2C N1(C(=O)Cn2nccn2)CC2CC1CN2C(c1cc(C2CC2)ns1)=O C1(CNC(Cc2ccn(CC)n2)=O)CCCN(C(C2CCC(C)O2)=O)C1 C(=O)(CC(C(F)(F)F)N(C)C1CC1)NCC1=CCN(C(C(F)OC)=O)CC1 c1(C2N(C(n3ccc(CC4CC4)n3)=O)CC2)nc(C2CC2)no1 c1(CC)nn(C)c(C(=O)N(C)CCNC(c2ocnc2C2CC2)=O)c1Cl N1(C(c2noc(C)c2C)=O)CCN(C(c2cc(Br)ccc2Cl)=O)C(C(C)C)C1 C(=O)(C(C)(C)CC(=O)N(C)C)N(CC(C)NC(=O)Cn1ccc(Br)n1)C N1(C(C2C(=C)C2C(=O)OC)=O)CCCC1(C(=O)N(CC(O)C1CC1)CC)CC C1(N(C(C(CC)SC)=O)C)CCCN(C(=O)CCc2cc(Cl)cs2)CC1 N1(C(CNC(C)=O)=O)CCC2CN(C(c3c[nH]cc(Br)c3=O)=O)CC2C1 CC1(CS(=O)(=O)NCc2cnoc2)COC1 c1(C(N2CCN(C(C(=Cc3cccnc3)C)=O)CC2)=O)nc(O)c(C#N)cc1C CCCCCCCCOCC(N1CCC(NC(c2snnc2C)=O)C1C)=O S(=O)(=O)(c1cc(C)cnc1N1CCC(c2ccncn2)CC1)N(CCSC)CC N1(C(C(=O)NCCC)C2CC2Cl)CCC(N(C)CC2CC2)CC1 c1(OCC(=O)NC(C)C(C)NC(=O)Cn2cccnc2=O)cncc(Br)c1 CS(=O)(=O)c1ccc(CNC(=O)CCNS(=O)(=O)c2cccc(Cl)n2)cc1 C12(NC(=O)CCc3cnoc3)CC(CNC(C3CC=CC3)=O)(C1)C2 Cc1nnc2n1CC(C(=O)NC13CC(NC(=O)CC4(CO)CC4)(C1)C3)C2 C1(n2cc(C(C)O)nn2)(C(=O)OC)CCN(C(=O)N(C)CC2(SC)CC2)CC1 CCC(CC)C(=O)NC1(C(=O)Nc2ccc(CO)nc2)CC1(C)C N1(C(C(C(C)C)O)=O)CCCCC12CN(C(=O)Cc1csc(Br)c1)C2 c1(CCC)nc(C(=O)NCC(O)CNC(C2CC(S(C)(=O)=O)C2)=O)co1 c1(C(=O)NCC2N(C(COCC(=O)NC)=O)CCC2)ccc(F)c(C)c1Cl c1(N(CCCOCC)C)ccc2cc(S(=O)(=O)N3CCC(C)(F)C3)ccc2n1 c1(SC(C)(C)C)ccc2c[nH]nc2c1.n12cc(nn1)NC(=O)N1CCC(C1)C2C Cn1nc2c(c1C(=O)NCC1CN(C(c3ccc(O)nn3)=O)C(C)(C)C1)CCC2 c1(C(=O)Nc2cc(-c3cn(CC)nc3C3CC3)[nH]n2)cc(Cl)c(Br)c(Cl)c1 C1(C(N2C(C(=O)OCC)CC2)=O)CC(C)(NC(=O)Cn2nccn2)C1 N1(C(C2CC(=C)C2)=O)CC(C2CCCCN(C(=O)CCC3C(=O)ON=C3C)C2)C1 C1(C(=O)NCc2cncc(OC)n2)CN(Cc2ccc(C)cc2Cl)CCC1O c1(C2C(C(=O)NC(CNC(CCNS(CC)(=O)=O)=O)C)C2)c(C)nn(C)c1Cl Cc1c(C(=O)NC(C2(O)CN(C(C3CC(CC(F)F)C3)=O)C2)C)ncn1C CCCCC(CN(C(=O)CC(C(F)F)NC(=O)CN1CCN(C)C(=O)C1)C)CC N1(C(C2=C(C#N)CCC2)=O)CCC2CCN(C(c3cc4ccncc4o3)=O)C2C1 Cc1cnc(C(=O)NCC2(O)CCCN(C(=O)Cc3nc[nH]n3)C2)cc1Cl C1(N(C(Cn2nnc(C)n2)=O)C)CN(C(=O)COCCN(C)C)CC12CC2 c1(C(=O)NC(C)CCCNC(=O)CCCC2CC2)n[nH]c2c1CS(=O)(=O)CC2 CCN=c1[nH]c(C)c(C(=O)NCCOCCn2cc(-c3ccc(C)s3)nn2)s1 C1(N(C(C2N(C(C)=O)CCC2)=O)C)CC2CC1N(C(C1CC(C)(O)C1)=O)C2 N1(S(C)(=O)=O)CCC2(C)C(C1)C2(Cl)Cl.C1CN=C(NC2CCCC2)NCC1 c1(C(N(C(C=C(C)CCC(N)=O)=O)CC(N)=O)=O)cc(C)ncc1C CC1(CCNC(C2(CNC(C3CC3Cl)=O)CCCO2)=O)CCOCC1 C1(OC)CCC2(C(=O)NCC3CN(C(=O)C(F)C4CCC4)CC3O)CCC12 Cc1nc2cc(C(N3CCCC(CNC(=O)CC4C(C)C4(F)F)C3)=O)cnc2[nH]1 N1(C(CCCCCCCC)=O)CCC(C2(O)CN(C(c3ccsc3Cl)=O)C2)CC1 C#CCC(O)C(=O)NCCC(C)NC(c1c(C)ncn1O)=O C1(CC(=O)N(CC(=O)OCC)CC#C)CN(C(C)=O)CC1C(F)(F)F C(=O)(C1CCCc2sccc21)N1CC(SC)C(NC(c2ccoc2Cl)=O)C1 C1(CC(=O)N(CC(C)(C)NC(=O)CS(=O)(=O)NC2CC2)C)CCCCC1(F)F c1(C(=O)OC)cc(N(C(=O)C=CCF)C)ccc1[N+](=O)[O-].C12(C)CCCC1NC2 C1(CNC(CC2CCC(C)C2)=O)CC2(CCC2)CN1C(=O)C=Cc1ccsc1 Cc1ccc(F)c2c1CN(C(c1cccc(Cl)c1C)C(=O)NC(C)C)CC2 N#Cc1ccc(=NC2CCN(C(C3COC4(CCC4)C3)=O)CC2)[nH]n1 C1(CC(=O)N(C2CN(C(c3cc(Cl)c[nH]3)=O)C2)C)CCCCC1O N1(C(c2c(C)nc(O)nc2C)=O)CCCC(C2CC2NC(c2ccoc2C)=O)C1 C1(CNC(c2c(C)noc2C)=O)CCC(C)CN1C(C12COC(CSC)(C1)C2)=O c1(C(=O)NCCCN(CCC)C(c2ncc(F)cn2)=O)ccc(=O)n2c1CCC2 c1(OC)c(C(N2CCCC(N(C(=O)C(F)CC(C)C)C)C2)=O)cccc1[N+](=O)[O-] c1(CC(=O)NC2CCCN(S(=O)(=O)C(F)(F)F)CC2)ccc2c(c1)OCCO2 n1(CC(=O)N(C)CC2CN(c3ncnc(=N)[nH]3)C2)nc2c(n1)CCCC2 N1(C(c2cc(=N)[nH][nH]2)=O)CCC(NC(=O)C2=CCSC2)C(CO)CC1 CC(CNC(=O)CNC(C1CC1(Cl)Cl)=O)CN(C)C C(=O)(CC(c1ccccc1)NC(N)=O)NCC(CN(C(=O)COCCCF)C)O C(=O)(C(C)(O)C(C)(C)C)NC(CC)CNC(=O)CCc1csc(C)n1 c1(OC)ncc(Br)cc1CN1CCC(F)(C(=O)Nc2ccc(O)cc2C)C1 c1(C2(NC(=O)Nc3c(CC(N)=O)csc3)CCCC2)ccccc1F C1(C(=O)NC2C(C)CCN(C(COCC)=O)C2)CCC(C2CCCO2)O1 C1(N(C(c2n(CCC(=O)OC)ncc2)=O)C)CCCN(C(=O)C(CO)OC)CC1 C(=O)(C(F)C(C)CNC(c1ccn(C)n1)=O)N1C(CC)C(O)CC1 c1(C(=O)NC(C)CNC(C2(CO)CC2)=O)ccnn1C(C)(C)C O=C(C1=CCCOCC1)N1CC(C(=O)NCCNC(C23CSCC2C3(F)F)=O)C1 c1(C(c2cscn2)NC(=O)NC2CC2CC2(CO)CCC2)ccccc1 C(C(CC(=O)N(C1COC(C)(C)C1)C)NC(C1(c2cc[nH]n2)CC1)=O)OC c1(CC)nc(C)c(C(=O)NCC2(F)CCC(NC(c3cc(Cl)cn3CC)=O)C2)s1 c1(C(C)(C)NC(=O)NC(C(C)N2CCCC2)C2CC2)ccccc1 c1(C(=O)NCCCCCNC(C2(n3cncn3)CC2)=O)sc(Cl)cc1Cl Cc1ccn(CC(=O)NCC2CCN(C(=O)CC3CCOC(C)(C)C3)C2)c(=O)c1 C(=O)(C1=NN2CCC(C)N=C2N1)N1CC(O)(C(C)NC(C(F)=C(C)C)=O)C1 c1(C(N2CCC(NC(C(COC)OC)=O)C(F)C2)=O)ccc2cc(O)ccc2c1 C#CC1CCN(C(=O)CC2CN(C(=O)C3=CCSC3)CC2C)C1 c1(C(=O)NCCN(C(C2CC(OC(F)F)C2)=O)CC)ccc(Cl)c(C)c1O C(=O)(C(CCC(N)=O)N(C)C)NC(C(C)C)C(=O)NC1CCNC(C)CC1 C=CC1(CC(=O)NCCN(C(=O)CN(c2ccncc2)C)CC)CCCCC1 CN1CCC(OCCN(C)C(C2(N(C(=O)CC3CCCC3)C)CC2)=O)CC1 C1(NC(=O)Cn2cc(Br)cn2)CN(C(c2ccccc2CO)=O)C2CC12 C1(NC(C2C(OC)CC2)=O)CC2CC1CN(C(c1cn3ncnc3nc1C)=O)C2 CCC(CCC(=O)N1CCN(C(C)=O)C(C)C1)NC(=O)CC(C)F C1(CNC(c2cc(CCCCC)[nH]n2)=O)C(C)CCN1C(c1c[nH]c(=O)cn1)=O C(=O)(CCCCC(C)C)N(C1CC1)C(C)Cl.C(CC(=O)N(C)CC)NC(=O)NC CCC(CC)CCC(=O)N(C(C)C(N1CCC(CC(F)F)C1)=O)CC c1(NC(N2CCC(CCNC(C3CCSC3)CC)CC2)=O)ccc(C)c(C)c1 CC(C)C(C(C)NC(c1ccccc1F)=O)NC(c1ncccc1C(F)(F)F)=O CC1(C(=O)N2CCC(C3(NC(=O)C4=CCCO4)CC3)C2)CCCc2ccccc21 C(CCC(C)(C)C(=O)NC1C=CCN(C(=O)CC2(C)CC2)C1)OC CC(C)C(F)C(=O)N1CCSCC1CCNC(C1COC(C)C1)=O N1(C(C2C(SC)CCC2)=O)CC(O)(C2CCN(C(C3(SC)CC3)=O)CC2)C1 N1(C(C)=O)CC(O)CC1C(N1CCCC(N(C(=O)C(C)(C)NS(C)(=O)=O)CCO)C1)=O C1(NC(=O)CC2COCC2O)CC12CC(NC(c1ccccn1)=O)C2 C1(NC(C=C(COC)C)=O)CC2CCC(C1)N2C(C1CC12CCOCC2)=O CC(F)(F)CCC(=O)N1CCCC(F)(CNC(=O)CC(O)C2CCCC2)C1 C1(NC(C(C)CN(C)C)=O)CC2(CCC(NC(=O)C(F)CC3CCCC3)CC2)C1 Cc1ncncc1C(=O)NC(C)C(C)(C)NC(C1CC(c2ccccc2)C1)=O N1(C(CC2ON=C(C)C2)=O)CCN(C(c2cc3n(n2)CC2(CC2)C3)=O)CC(C)(F)C1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)N(CC(O)CN(C(=O)C#CC(C)C)C)C c1(CC)ccc(C(N2CCC(C)(CNC(C34CC(F)(CO3)C4)=O)C2)=O)nc1 N1(C(C2N(OCC)CCC2)=O)CC(C(=O)NC)CC(C)C1 CN1CCCC(c2cn(CCCc3nc(CCc4cccnc4)no3)nn2)C1 C12(C(=O)NCc3nc(C)c(C)o3)CCCC1CCN2C(C1CC(N(C)C)C1)=O N1(C(c2c(C)n[nH]c2)=O)CC2(C1)CN(C(=O)C(C)(C)CN1CCOCC1)C2 N1(C(C(CC2CN(C(C(CC)OCC)=O)C2)F)=O)CCC(O)(CC)CC1 C1(C(=O)NC2(C)CCCO2)COCCN(C(=O)COC2CC2)C1 CC1(CNC(C2C=CCCN2C(C2CC(CC3CC3)C2)=O)=O)CCC(O)CC1 N1(C(c2ccnn2C2CC2)=O)CCC2CC2(C(=O)NCc2nncs2)CC1 C1(C)(CNC(C=C(C)Cl)=O)CCCN(C(=O)Cc2ncccc2C)C1 C(=O)(C(F)(F)C1=CCOCC1)N1CC(CNC(C(C(C)C)O)=O)C2(C1)CC2 NS(=O)(=O)CCCNC(C1CC1c1cn(CCc2ccc(O)cc2)nn1)=O Cn1nc(C(=O)NC(CO)CCCNC(c2cncc(N)n2)=O)cc1F C1(N2CC(CN(C3CCC3)C(=O)OC(C)(C)C)C2)CCC2(CCC2)O1 C1(N(C(COCC(C)C)=O)C)CCN(C(c2n[nH]c3c2CCC3)=O)CC12CC2 C(C(C)(O)C(C)C)NC(C1C(CNC(COC)=O)CCC1)=O N1(C(=O)C(C2CC(F)(F)C2)O)CCCC12CCS(=O)(=O)CC2 C123CC4CCC(C1C2)N4CCN=C1N=C3C=CN1.N1(CC2CC2)CCCCC1 C1(NC(c2cc(C3CC3)[nH]n2)=O)CN(C(=O)CCc2cc(Br)cs2)CC1O N1(C(COCCC)=O)CCCC(O)(CNC(=O)COC2CCCCCC2)C1 C(=O)(CCCCCCc1c[nH]c2ccccc12)NC(CNC(C(C=CC)O)=O)C CC1(NC(=O)CC2CC2(Cl)Cl)CCN(C(=O)CC23CC(C2)C3)C1 c1(C(=O)NCc2nc(CNC(C(CSC)O)=O)sc2)ccnc(C)c1 NC(=O)CCCCC(=O)NCCCOCCC(N1CCCC2(CC1)CC2)=O N1(C(CC2C(C)OC(C)C2)=O)CC2(COC(COC(C3(C(=O)N(C)C)CC3)=O)C2)C1 C(C)(C(C(=O)N1CCCCC1C(=O)NCc1nc(C)c(C)[nH]1)N(C)C)OC N1(C(C(=O)NCC)=O)CCCC12CCN(C(=O)CC1CCCO1)CC2 C1(C(=O)NCC(C)(C)OC)CCC(C(C)C)N1C(=O)C=Cc1ccc[nH]1 Cc1ccc(C)c(CC(N2CC(C(=O)Nc3cc(Cl)nnc3Cl)CC(F)C2)=O)c1 C(=O)(C1=C(C#N)CCC1)NC(C1CCCCC1)C(=O)NCC(C(C)(C)O)F C1(NC(C2C(OC)CCC2)=O)CN(C(c2cnccc2N(C)C)=O)CC1C(F)F C(CC(O)C(=O)NCCC(=O)NC(c1csc(C)n1)C)SC C(=O)(CC(C)(C)CNC(c1cc(C)nc(O)n1)=O)N1C(C)CSCC1 C1(C(=O)NCC(C)CCl)CCCC12CCN(C(c1cc(F)c[nH]1)=O)C2 c1(C(N2CC(n3cc(-c4ccc(C#N)s4)nn3)(N(C)C)C2)=O)ncncc1C c1(C(=O)NCC2(F)CCN(Cc3c(F)cccc3F)C2)cc(Cl)cnc1O c1(C(N2CC(NC(c3c(C)nn(CC)c3C)=O)C(C)C2)=O)cc(F)cc(Br)c1F c1(C(=O)NCC2CC(NC(c3c(CC)oc(C)c3)=O)C2)nc(C)ccc1Br C1(COC)(NC(c2cncc(SC)c2)=O)CCCN(C(c2c[nH]c(=NC)s2)=O)C1 N1(C(Cn2ccc(C)n2)=O)CCC(NC(c2cc(C(F)F)ccc2F)=O)C(F)C1 C(=O)(N=c1cc[nH]cc1)OC.c1(C2C(=O)N2C2CCC2)cccc(Cl)c1 c1(C(N2CCN(C(c3ccc(O)cc3)=O)CC2CF)=O)ccc2ncccn12 C=C(C)CC(C(=O)NCC(CC)(CC)NC(=O)Cc1ccn(C)n1)OC Cc1c(CN(C)C(C2CC(C)N(C(=O)C=CC(C)(C)C)C2)=O)cnn1C CC(C)CCC(F)C(=O)NC(C)(C)C=CC(=O)NCC1COCC(=O)N1C C(=O)(C1NCc2nc(C)ncc21)CCN(C(C1OCC(C(=O)OC)C1)=O)CCO C(=O)(C1=NNC(=O)C1)N1C(CN(C(C(CCC)N(C)C)=O)C2CC2)CCC1 C1(c2nc(CNC(C3C(C(C)C)C3)=O)[nH]n2)CCN(C(C23CC(C)C2C3)=O)CC1 c1(C(=O)NCC(C(C)(C)C)NC(C2N(CCC)C(=O)CC2)=O)cc(F)ccc1C C(C(C)(CO)NC(c1cn(C2CC2)nn1)=O)NC(CN1CC(C)C1)=O N1(C(C(C2CN(C(C=CC(C)C)=O)C2)O)=O)CCC2(CC=CCO2)C1 C1(NC(C(C(C(C)C)O)C)=O)CN(C(=O)C2=C(Cl)CCC2)C2(CCOCC2)C1 C(=O)(CS(=O)(=O)C1CC1)OC.C12CC(C3CC13)OCC(=O)NOC2 C12(NC(c3cnc(C)o3)=O)CCCC1CN(C(=O)Cn1cc(C3CC3)cn1)C2 c1(C(=O)NCC2C(NC(c3c(CC)c[nH]n3)=O)CC2)cc(-c2ccco2)ccn1 n1(-c2ccn(CCOCC)n2)nc(-c2cccc(F)c2)nc1C(C)OC N1(C(C(CC)(C)O)=O)CCC2(CC1)CN(Cc1ccc(O)cc1OC)C2 Cc1cc(N)cnc1C(N1CC2C(N(C)C(C3CCC(=O)NC3)=O)C2C1)=O Cc1nc(C2CC2)oc1C(=O)N(C(C)CCNC(c1ccoc1Cl)=O)C c1(C(=O)NCC(C)(C2CC2)NC(c2cnc(S)[nH]2)=O)csc(CS(C)(=O)=O)n1 Cn1ncnc1CCC(=O)NCCCN(C(=O)CCCC1CCC1)C1CC1 C(C(CN=C(NC)NC1CCCC1)C(C)C)O.C1(CNS(C)(=O)=O)CCCC(CC)C1 N1(C(CN(CCCN(C)C)CC#C)=O)CCN(C)CC1 c1(C(=O)NCC2CCC(C)CN2C(=O)CN(S(C)(=O)=O)C)coc(S(N)(=O)=O)c1 c1(C(N2C(CN(C(C3C(=C)C3)=O)C)CCC2)=O)cnc(C)c(C)c1 N1(C(CC2CCC(C)(C)C2)=O)CCCCC(C(=O)NCC2CC3(C2)CC(O)C3)C1 C1(CNC(CCC#C)=O)C(C2CC2)CCN1C(=O)C=Cc1c[nH]c(=N)c(C)c1 CC(O)(CNC(c1sccc1C1CC1)=O)CNC(C1CC1c1ccco1)=O Cc1ccc2c(c1)CC(C(=O)N(CCCCNC(=O)C(F)OC(F)(F)F)C)S2=O C(CCN=c1ccc(C(F)(F)F)n[nH]1)Oc1c(F)ccc(C)c1 N1(C(c2c(C)ccnc2)=O)CCC(C2(NC(C3CCC(CCO)CC3)=O)CC2)C1 CCCCC(O)C(=O)NC1CCN(C(c2cn(CCN(C)C)nn2)=O)C1(C)C CN1CCC(COC(C2(c3cncn3C)CC2)=O)CC1 N1(C(c2ccn(CCC)c2)C(=O)NC(C)C)CCCC(COCC)C1 CC1(C)CC(NC(c2cnc(CC3CC3)s2)=O)CCN(C(=O)CC2=CCCC2)C1 C(C(COC)CC(=O)N1CC(C(=O)N(CC(C)O)CCO)C(C)C1)OC N1(C(C(CC=C)CC)=O)CCN(C(=O)C2=CCCCCC2)C2CS(=O)(=O)CC12 C(CC)(C(=O)NCC#CC(=O)N1CCCC1C1(C)CC1)OCC CCCCC(CNC(=O)C=C(Cl)Cl)NC(=O)C(O)COCc1ccccc1 c1(C(N(C(C(=O)NCC(C)C(F)F)C2CC2)C)=O)ccc(O)nc1 c1(OC)cncc(C=CC(=O)N(CC(C)N(C(=O)CCCn2ccnc2)C)C)c1 N1(C(c2cc(Cl)n[nH]2)=O)CCCc2cc(-c3ccccc3F)ccc21 CCC(CC(C)C)C(=O)NCC1(CNC(=O)C(C)CC2CCC2)CCC1 c1(C(=O)NC2(C(NOC(C=C)C)=O)CCSC2)ccc(C)n1C Cn1nnc(C(=O)NC2COCC2CNC(=O)CCc2cccc(F)c2)c1N CC(C)(C)C(=O)C(=O)N1CC=CC(C(=O)NOCCC2CC2)C1 C=C(Cl)C(C)(C)C(=O)N1CCC(O)(CNC(C2CCCCO2)=O)C1 C1(COC)(NC(c2c(Cl)ccnc2C)=O)CCCN(C(c2cccc(N)c2)=O)C1 C1(NC(c2c(CC)ncs2)=O)CCOCC1NC(=O)CSc1nnnn1C1CC1 C1(CNC(c2c(CC)c[nH]c2)=O)CC(NC(=O)CCCc2cncs2)C(O)C1 N1(C(C2N(CC)CCCC2)=O)CCCC2CN(C(=O)CCCSC)CCC12 c1(C(N2C(C)CC(NC(COCCC=C)=O)C2)=O)c(Br)nc2n1CCOC2 C1(NC(c2c(CC)cns2)=O)CN(C(=O)C(C)(C)c2ccno2)CCC1C C(=O)(C(C)(C)C(=O)NC(C)CCCNC(c1ccccc1OCC(F)F)=O)OC C1(OC)CCC(C(=O)NC2CC(CN(C(C3(C)CC3C)=O)Cc3ccccc3)C2)C1 CCC(CC(=O)N1CCC(CC)C1CNC(c1cnncc1O)=O)C1CCC1 Cc1cccc(F)c1N(C(=O)CONC(=O)CN1C(C)CCC1C)C1CC1 n1(CC(=O)N(C)CC2(NC(CSSC)=O)CC2)ncccc1=O c1(OC)ccc(C)c(C(=O)N(C)CC2CCN(C(=O)C(C)S(C)(=O)=O)C2)c1N C1(C(=O)NCC(N2CCSCC2)C)CN(C(=O)C2CC2)CC12CC2 c1(CC)cc(C(N2CCSCC2C(=O)NC2(CCO)CCC2)=O)c(C)o1 C1(CC(=O)NC(CCNC(C2OCCN(CC)C2)=O)(C)C)CCn2cncc2C1 C1(n2cccn2)(C(=O)NCCC(C)CO)CCN(C(=O)CC2CC3(CCC3)C2)CC1 C1(C(=O)NCCOCCNC(C(CC=CC)C)=O)CCC(F)(F)CC1 c1(C(=O)OC)cc(Cl)c(NCC2CC(C)N(C(c3[nH]c(C)nc3C)=O)C2)nc1C C#CCCCCC(=O)N1CC2(C)CC1(C(=O)NCCOC1CCOC1)C2 c1(N2CCN(C(c3c(C)c[nH]n3)=O)CC2)ncnc(C)c1C#N C1(CNC(c2ccc(CCO)nc2)=O)CC(=O)NC(=O)C1.C12(CCC1)C(=O)NC2 Cc1nncc(C(N2CCC2CC(N2CCC3(CCC3)C2)=O)=O)c1C c1(CNC(CC(CCC)NC(C2(COC)CCC2)=O)=O)ccc(C#N)cc1C C1(NC(c2ccc(OC)o2)=O)CN(C(=O)Cn2cc(N(C)C)nn2)CCC1C N1(C(C2N(C(C(C)C(F)F)=O)C3CCC2C3)=O)CCCC(C)(O)CC1 c1(C(=O)NCCOC(C)(C)CNC(=O)C2=COCCC2)ccc(C#N)nc1O N1(C(CC(CC)C)=O)CCCCC(CCC(=O)NC(c2ccc(F)cc2)C)C1 c1(OC)cccc(C(=O)NCC(CO)NC(=O)CCc2ncccc2C)c1 N1(C(C(=O)NCC(F)(F)F)=O)CCCC2(NC(C3(c4ccccc4)CC3)=O)CC12 c1(C(=O)NC(CNC(C2(C=C)CC2)=O)CCC)onc2c1CCCC2 C1(CNC(=O)Cn2cc(Cl)cn2)C2CN(C(c3cnncc3O)=O)CC12 C#CCCCC(=O)NCC(c1ccc(C)cc1)NC(C1(C)COC(=O)N1)=O c1(C(N(C(c2n(C(C)C)ccn2)C(=O)NC2CCOC2)C)C)cccc(Cl)c1 Cc1cc(O)c(Cl)cc1C(=O)NC1(CCCNC(C2C=CCCC2)=O)CC1 C(c1cccnc1)=C(C(=O)NC(CC)C(=O)OC)C CC1(CNC(C2(C)C=CCCC2)=O)CCN(C(=O)Cc2ccc(O)cn2)C1 C1(NC(c2ccc(F)cn2)=O)CC(O)CN(C(=O)CCC=CBr)C1 c1(C(=O)NC2C(C(=O)Nc3ccnc(OC)c3F)CCC2)ccc(O)c(C#N)c1 c1(C(=O)NC(C)CCCNC(c2ccc(O)cc2F)=O)ccc2c(c1)C(=O)OC2 Cc1cccc(NC(=O)C(=O)NCCN(C2CC(Cl)(Cl)C2)C)c1 C1(C)(CC)CC(C(=O)NCC(C2CCNCC2)(C)C)CCO1 C1(CC(=O)NC2(CCC(=O)NC(C)Cc3nncn3C)CCC2)CC2C=CC1C2 N1(C(c2c(OCC)cccc2)=O)CCCCC(NC(=O)C=C2CCSCC2)CC1 N1(C(c2n(CCCC)ncc2)=O)CC(C)C(C)(CNC(=O)CCOCC(C)C)C1 C1(C(N(CCSC)CC)=O)C(C2CC2)CCN1C(c1cc([N+](=O)[O-])n[nH]1)=O N1(C(CC(C)c2ccco2)=O)CC2(CC(CNC(c3cnc(C#N)s3)=O)C2)C1 C1(NC(c2nn(C)c(O)c2)=O)CCN(C(C23CCCC2C3(F)F)=O)CCC1(F)F Cc1cc(N)cnc1C(=O)NCCC(C)(C)C(=O)NC1CC(n2cncn2)C1 N1(C(C=Cc2cc(C)no2)=O)CCN(C(C2CCCN2C(C)C)=O)CC1CCO C1(CN2CC(Oc3c(Cl)ccc(C(=O)OCC)c3)C2)CCC2CCCC2O1 N1(C(C(C)NC(=O)NCC)=O)CCCN(C(C2(SC)CCC2)=O)CC1C C1(CN(C)C(C2(CNC(=O)CC(C)(C)O)CCCCC2)=O)C(C)(C)C1(C)C c1(SCC(=O)NCC2CCC2)ccc(C#N)cc1.C12(CCCCC1)C(=O)N2.CC Cc1cc2[nH]c(C(=O)NCCC3CCCN3C(=O)CC(C)(O)C3CC3)cc2o1 N1(C(c2cnc(C3CC3Cl)s2)C(=O)N(C2(C)CC2)CCC)CCC(O)(C(C)(C)C#N)C1 C1(C(=O)NCCCCC(C)NC(=O)COCc2cccnc2)CCCC1C1CC1 c1(C(=O)NCC(CNC(C2C(c3c(C)c[nH]n3)C2)=O)O)coc2c(C)cccc12 O=C(CCN=C(NCc1cccs1)N1CCC(NCCF)C1)N1CC1 N1(C(C=C2CCN(C)C2)=O)CCC(NC(c2cc(C(F)F)no2)=O)C(C)(C)C1 CC1CN(C(c2ccnc(O)c2)=O)CC(C)CN1C(C1CC(=O)NC1(C)C)=O c1(N2CCCC(CNC(C3C(CCC)CCC3)=O)CC2)nc2cccnc2s1 N1(C(CC2CN(C)C2)=O)CCCC1CCNC(=O)Cn1cnnn1 c1(OCCC(=O)NC(CNC(C2(n3ccnn3)CC2)=O)CO)cccc(Cl)c1Cl C1(CC=C)(NC(=O)CC(=O)NCC(F)(F)F)CCN(C(C2CCOC2)=O)C1 c1(C(N(CCCCN(C)C(C2CCC(O)C2)=O)C)=O)[nH]nnc1-c1ccccc1 C1(C(N(CCC)CCO)=O)CC(C)N1C(=O)Cn1cnc(=N)[nH]1 N1(C(C(C(C)C)O)=O)CCC(C)N(C(=O)C(=O)NCCC(N)=O)CC1 c1(C(=O)NC2CCC(NC(C(N(C)C)C3CC3)=O)CC2)c[nH]c2ccc(F)cc12 c1(CN(CCOC)C(c2ccccc2)C)ccc(Cl)cc1 CC(C)(CNC(=O)CNC(N)=O)CCNC(c1cccc(-c2ccoc2)c1)=O C(=O)(CN=c1cc[nH]cc1)NCC(C)N(C(=O)C(CO)C(C)(C)C)C c1(CCC(=O)NCCC2(NC(CN(CCC)C)=O)CCCC2)ccc(F)cc1F CC1OCCN(C(c2ccncc2)=O)C1C(=O)NC1CC(CCO)C1 CCC(CN=c1nc(N(C)Cc2conc2C2CC2)c2sccc2[nH]1)C(C)(F)F c1(CS(C)(=O)=O)n[nH]c(=NC(=O)NCC(c2cccc(O)c2)CO)s1 c1(C(=O)OC)ccc(CNC(N2CCCCC2C2CCCC2)=O)c(C)c1 C1(NC(C(C)NC(=O)NC)=O)CCSC12CN(C(c1scnc1C(C)(C)C)=O)C2 N1(C(CNC(CSSC)=O)=O)CCC(N=c2[nH]nc(CC)o2)C(CC)C1 c1(CNC2CCC(NC(C3C(OCC)CC3)=O)CC2)cc(CC)cc(OC)c1O c1(CCC(=O)NC(CN(C(=O)Cc2ccoc2)CC)C)cccc2c1OCO2 CCCCCCC(C)C(=O)N1CC(C(N2CCC(n3ccnn3)C2)=O)C(CC)C1 C1(c2onc(C)n2)CCC(c2cn[nH]c2)(NC2CC2CC(C)C)CC1 CCC(C)CC(C(=O)N(C)Cc1ccc(C)cc1)NC(c1cc(C#N)c[nH]1)=O c1(C(CNC(=O)CCSC)NC(c2c(CC)nco2)=O)ccccc1OC CN1CC(=O)Nc2cc(C(=O)Nc3ccc4c(c3)CCC4)ccc21 C1(CNC(CCSC)=O)CN(C(=O)C(C)c2cc[nH]n2)C2CCCC2O1 C1(CC)COC(c2ccccc2)CN1CC(=O)NC N1(C(CC2CCC(=O)N2)=O)CCC2CN(C(c3ncc(Br)cn3)=O)C2C1 N1(C(C(=Cc2ccco2)C)=O)CC2CC(C1)CN(C(c1ccc(C(N)=O)[nH]1)=O)C2 CC1CN(C(=O)CC(C)n2cccn2)CC1CCNC(C1CC(O)C1)=O C1(CCNC(C(C)SC)=O)CC(F)(F)CN1C(=O)COc1cccc(C(C)C)c1 N1(C(C2CN(C(c3c(C)cco3)=O)CC(F)C2)=O)CCc2ccccc2C1 CC1OC2(C)CC1(C(N1CC3CC1CC3NC(=O)CN1C(=O)C(=O)NC1=O)=O)C2 CCC(CC)(CC)C(=O)NCC1(NC(c2cc(O)ccc2Br)=O)CC1 C(=O)(N1CC(C)(O)CO1)C1(NC(CCC(C)N(C)C)=O)CCN(C)C1 C1(NCCC(=O)Nc2cccc(OC)c2)CN(C(=O)C(F)(F)F)CC(F)(F)C1 S(=O)(=O)(C1CCOCC1)NCC1N(C(C(C(C)C)O)=O)CCCC1 c1(C(=O)NCC(CC=C)NC(=O)Cc2cscn2)cnc2c(cnn2C)c1N N1(c2nc(=NC)nc(N3CCC(C(CC)CC)C3)[nH]2)CCC2(CNC(=O)N2)C1 C1(C(=O)NCC#CC(=O)NCC(C)C2CC2)C2CC3C(C2=O)C13 c1(C(N(C)CC2CCN(C(C3(C)CCCN3C)=O)C2)=O)nc2ncccn2n1 N1(C(C2(CC#N)CCCC2)=O)CCOC(C(=O)Nc2ccc(O)cc2)C1 N(C(=NCCN1CCC(C)C1)NC1C(C)(C)C1(C)C)CCOCC N1(C(C2C(CCC)C2)=O)CC2CCC1CN2C(C1(OC)CCSC1)=O C1(C(N2C(C)CCC(NC(C3CCC(=O)N3)=O)C2)=O)CCc2c(nnn2C)C1 C#CCC(O)C(=O)N1CCCC1(C)CNC(c1ccc(C2SCCS2)cc1)=O c1(CCNC(CN(C)C(N)=O)=O)ocnc1CNC(=O)CCc1cnn[nH]1 c1(C(=O)NC2CN(C(c3cnn(CC4CC4)c3)=O)CC2F)ccc2n[nH]cc2c1 C#CCC(C)(C)C(=O)NCCCNC(=O)C(C)Cc1ccc(Cl)c(Cl)c1 C(CCCCCCO)n1cc(C2CCCN(C(C(=O)OC)c3cscn3)C2)nn1 C(=O)(C(C)(C)CC(=O)N1CCC(O)(CCNC(=O)CN2CCCNC2=O)C1)OC N1(CC)CCCC1CC(=O)NCC(O)CCNC(C1(n2ccc(CC)n2)CC1)=O Cc1cc(C(=O)NCCC(C)NC(=O)Cc2cncs2)nc(Cl)c1 C1(CC(=O)NCC(CN(C(=O)CC2COC(=O)C2)CC)(C)C)CCN(C(C)=O)CC1 C1(CCCCNC(c2ccc(C(F)F)nc2)=O)CCCN(C(=O)C(F)(F)CO)C1 c1(C(N2CCCC(CN(C(CC(CCC)O)=O)C)CC2)=O)ccc(Cl)c(Cl)c1C c1(CCC(N2CC(O)CC2CNC(C2(C3CC3)CC2)=O)=O)ccc([N+](=O)[O-])cc1 CC1C(NC(c2cc(-c3ccco3)on2)=O)CCCN1C(C1CS(=O)(=O)C1)=O C1(CNC(c2onc(CC)c2C)=O)CN(C(C2CN3CCC2C3)=O)CCCO1 c1(CN=C(NC2(C=C)CCC2)NC(C)COC)cc(C)nc(O)c1 CC1=C(C(=O)NCC2(F)CC(CNC(=O)CC3CCCC3C)C2)CC1 C1(CCNC(C=CC(=O)OCCC(N)=O)=O)CCCN1C(=O)Cc1cccs1 c1(C(=O)N(c2ccccc2)C2CN(C)C2)ccc(-c2cccc(C3CC3)n2)cc1 N1(C(C(c2c(C)cccc2)C)=O)CC2CC1CC2NC(=O)CSCCN(C)C C1(C(=O)NCC2CC(NC(c3cccc(F)c3)=O)C2)C2CCCCCCC12 C1(NC(CC(CC)SC)=O)CCC2CC1CN2C(C1(C#N)CCOC1)=O c1(N2CCC(C(C)NC(C3CCN4CCCC4C3)=O)C2)nc2cccc(N)c2s1 N1(C(C=NOC)=O)CC2CCN(C(c3cc4scnc4[nH]3)=O)CC12 CC(CC(N)=O)C(=O)NCC1CCN1C(c1cc(-c2ccc(O)cc2)on1)=O C1(C(=O)N(CCCn2cc(Cn3cccn3)nn2)CC2CC2)CCC(F)C1 C1(CCNC(c2c(C)nc(CO)s2)=O)CN(C(=O)CNC=O)CCS1(=O)=O N1(C(C)=O)CCOCC1C(N1CCC(C)(CNC(=O)C2=CCC2)C1)=O C(=O)(CS(=O)(=O)CCO)N1CC(OCCNC(c2ccc(N)cc2F)=O)C1 C1(CNC(C2CN(c3nncs3)C2)=O)CC2CN(C(C3(Br)CC3)=O)CC12 c1(C(=O)NCC(C)(C)CO)n[nH]c2c1CCN(Cc1cc3c(cc1Br)OCO3)C2 Cc1nc(C)c(C(N2CCC(C(C)NC(C3CCCC(C)C3)=O)C2)=O)c(C)n1 c1(C(N2CC(CCNC(CC=C)=O)OCC2)=O)ccc2cc[nH]c2c1 Cc1cc(C(=O)NCc2nc(C(N3CC(O)CC3CN(C)C)=O)co2)cnc1O c1(CC)occ(C)c1C(=O)N(CCCN(C)C)CCNC(=O)CN1CCSCC1 C12(NC(C3CN(C(CCNC(=O)OCC)=O)C4C3C4)=O)CCC(CO)(CC1)CC2 N1(C(=O)OCC)CC(C(=O)N(CC(C)NC(=O)Cc2ccsn2)C)C1 c1(C(=O)NC(C(C)NC(=O)C=CCO)(C)C)ccc(S2(=O)=NCCC2)cc1 Cc1cc(C(N2CCC(NC(=O)C(C)(Cl)Cl)C(CO)C2)=O)cc(N)c1Cl C1(CCCNC(C(C)C2CCC2)=O)CCCN1CCc1ccc(-c2cc[nH]n2)o1 O=C1CC(C2CCCO2)(C(=O)NCCC2(NC(=O)CO)CC2)C1 c1(OC)cccc2c1OCCCC2NC(=O)C(=O)NC(CO)C(C)C N1(C(C)=O)CCCC(C(N2CCC(NC(c3cn(CCCF)nn3)=O)C2C)=O)C1 c1(C(N(C2CC23CC3)C)=O)nc(Br)cnc1N.CCC1CC(=O)N1 c1(C(N2CC(F)(C(N3CCN(C(C)=O)CC3)=O)C2)=O)cc(C#N)[nH]c1C c1(C(=O)NCCC2(NC(=O)CC3(O)CC3)CC2)csc(C(F)(F)F)c1 N1(CCC(N2C(C(N(CC(C)(C)C)CC)=O)CC2)=O)Cc2ccccc2C1 C1(CC(N2CC(C(N)=O)C2)=O)C2CCCC2N1C(C1(O)CCCCC1)=O c1(C(=O)NCC2(O)CN(C(C3(O)C(C)(C)C3)=O)C2)cccc2c1OCCN2 c1(C(N2C(C(=O)NC(C(C)C)CO)CC(C)C2)=O)cc2cc(Br)ccn2n1 N1(C(C(c2scc(C)n2)(F)F)=O)CC2(C1)CN(C(c1ccnc(C3CC3)n1)=O)C2 C1(NC(C2CCCN(CC)C2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CCC1CO c1(C(=O)NC2C(C)N(C(c3cnnc(O)c3)=O)CC2)ccc2c(c1)CCOC2 N1(C(C2CC(=C)C2)=O)CCC(F)(C(=O)Nc2ccc(CO)cc2F)CC1 C1(CN(C(C=CC)=O)CC)CCCN(C(=O)C(C)CCC)C1 C1(CC)CCC(C(=O)NC2C=CC(CNC(=O)CSCc3ncc[nH]3)C2)CC1 CN1N=C(C(=O)NC2(CNC(=O)CC3CC(F)(F)C3)CCCC2)CCC1=O c1(C(=O)OC)cc2[nH]ccc2cc1NC(c1cccc([N+](=O)[O-])c1F)=O c1(OC)csc(C(=O)NCC(C2CC2)N(C)C(C2C=CC=CC=C2)=O)c1OC C1(C(=O)NC(CCCC)CNC(=O)CCC(=O)NC2CCCC2)CCCS(=O)(=O)C1 C1(c2cn(CC3CC(C)OC3)nn2)CC(C)(C)OC1(C)C Cc1cnc(C(=O)NC2CCC(N(C(=O)C(C)n3cccn3)C)CC2)c(F)c1 c1(C(C)C(=O)N(C)CCOCCNC(C2(F)CCOC2)=O)cccc([N+](=O)[O-])c1 Cc1cc(-c2ocnc2C(=O)NCC2CCN2C(c2n[nH]c(C3CC3)n2)=O)on1 C1(NC(CCC(=O)OC)=O)CC2CCC1CC2NC(=O)CCOC(C)C c1(C(=O)NCC(CO)NC(c2[nH]n(C)c(=O)n2)=O)c[nH]c2cccnc12 N1(C(C2C(C=C)CC2)=O)CC(NC(c2snnc2C(C)C)=O)CC(C)(C)C1 C(=O)(C#CC1CCCO1)NC1C(CO)CCN(C(CN(C)C2CC2)=O)C1 c1(CCC(=O)NCC2(C(=O)O)CC2)ccc2nc(Br)sc2c1 c1(C(=O)NCC(C)CNC(C2CC2(C)C)=O)ccc(S(=O)(=O)N2CCCCC2)o1 N1(C(C(CC=C)(C)C)=O)CCC(C2CC2)(CNC(C2(OC)CCOCC2)=O)C1 C1(O)(CCNC(c2nc(C)sc2)=O)CCN(C(=O)Cc2ccc(O)cn2)C1 c1(OC)c(O)cc(C(=O)NC(c2ccc(O)nc2)C)cc1C#N C(N=c1[nH]cnc(NC(C2CCCCCC2)c2ccccn2)c1C)c1c(C)n[nH]c1 C(C)(CCN=C(NCc1c(C(C)C)cccc1F)NC(C)C)OC C(=O)(C#CC1CCCO1)C(C(C)C)CNC(=O)C(=O)NCCC(F)(F)F c1(C(C(=O)NCC2(F)CC(CNC(C3CC(=C)C3)=O)C2)O)ccccc1Cl N1(C(CC2(CSC)CC2)=O)CCC2CN(C(c3cccc(NC(N)=O)c3)=O)C2C1 c1(C(N2CCC(OCCC(=O)OC)CC2)=O)cc(Br)c(C)cc1Br C1(SC)CCCN(C(=O)C(C2CCN(C(c3cc(=O)cc[nH]3)=O)C2)F)C1 Cc1cccc(C(=O)NC(C2CN(C(c3ccc(OCCF)cc3)=O)C2)C)c1C N1(C(CC)=O)CC2CN(C(c3n[nH]c4c3CCC4)=O)CC2(C)C1 c1(C(=O)NC2CCC(NC(=O)COC3CCCOC3)C2)nc2cnccc2s1 N1(C(C(c2c(C)noc2C)OC)=O)CC(CNC(=O)C=C2CCC2)C2(CCC2)C1 C=C(F)C1(CC(N2CCCC2C2(C(=O)NC3CC(=O)N(O)C3)CC2)=O)CCC1 C(C(C)(C)CC(=O)N1CCCC1CF)NC(C1(C#N)C(C)C1)=O c1(CC(N2C(C(C)NC(C3CC3OC)=O)CCC2)=O)ccc(OC(F)F)cc1 N1(C(C(C2CC2)OC)=O)CC2C=CC1C(C(=O)NCc1ccccc1Cl)C2 c1(N2CCC(C#N)C2)nc2c(c(=NC3CCC4CCCC3O4)[nH]1)CCC2 N1(C(c2n(CC)ncc2)=O)CCN(C(c2cc3ccncc3o2)=O)CC12CCC2 N1(C(C(C(C)O)N(C)C)=O)CC2CCN(C(=O)Cn3nc(O)ccc3=O)C(C2)C1 CC(CNC(=O)CSC1CCCC1)(CO)NC(=O)CC=CCc1ccccc1 c1(CCNC(=O)Nc2nc(C(=O)OCC)c(CC)s2)ccc(F)c(F)c1 C(CN=c1nc2c(cnn2C)c(NCCc2n[nH]c(=N)o2)[nH]1)OCCOC CC1(C(N2CCCCC2CCNC(C2CCCC2CF)=O)=O)CCOCC1 c1(COC(c2cnc(C(=O)OC)s2)=O)ccc(C)nc1Br Cc1cc(C(=O)N(CC(O)CNC(c2cc(CO)n(C)n2)=O)C)[nH]c1C C1(C#C)(NC(C2(CC#C)CN(C(c3coc(SC)c3)=O)C2)=O)CC2CCCC12 N1(C(c2c(C)oc(C(=O)O)c2)=O)CCCC2CCCCCC12 CC1=NC(Cl)(C(C)C)C(N(C)CC2(CNC(c3cc(Cl)cn3C)=O)CC2)=N1 C(C(C)N=c1[nH]c2ncnc-2c(C(F)(F)F)[nH]1)NC(=O)NC(C)C N1(C(c2c(CC)cc[nH]2)=O)CC(NC(c2ccc(C(N)=O)[nH]2)=O)C(CC2CC2)C1 Cc1cccc(SCC(N2CC(OCCNC(C3CC3F)=O)C2)=O)c1 c1(C(=O)NC2CN(C(c3ccc(COC)[nH]3)=O)C(C)C2)cc(C)cc(Cl)c1 N1(C(c2c(C)cn(C)c2)=O)CCC(F)CC1C(=O)N(C)CC1CCC(=O)N1 C12(C(N(CCNC(CN3C(C)CCC3)=O)C)=O)CCC(CC1)C2(C)C N1(C(c2ccn(C)n2)=O)C(CNC(c2[nH]nnc2C2CC2)=O)CC2CC12 C1(F)(CNC(CCNC(COC)=O)=O)CN(C(=O)CC2CCC(C)O2)C1 c1(C(=O)NCC(C)(C)OCCNC(c2c(C)cc[nH]2)=O)c(C)noc1C(C)C N1(C(c2ccc(CNC(C(CC(C)C)OC)=O)o2)=O)CCC2CCCC2C1 C1(NC(CCCc2ccc(C)s2)=O)COCCN(C(C23CCCN2CCC3)=O)C1 N1(C(C2(F)CCN(C(C(C)NC(=O)OC)=O)C2)=O)C2CCC(C(N)=O)C1CC2 C1(CNC(=O)C=CC=C(Cl)Cl)CC12CCN(C(C13CCCN(CCC1)C3)=O)CC2 C(=O)(C(C)C(O)C(C)C)N1CCC(C(=O)N(C2CCN(OC)CC2)C)(OC)C1 C(=O)(C#CC(C)(C)C)NC(CC)CNC(c1cn(-c2ccccc2)nc1C)=O c1(CC)cc(C(=O)NCCC(C)N(C)C(c2cncc(N)c2)=O)cc(Cl)n1 C1(NC(CC(=O)OCC)=O)CCN(C(c2c(C(F)(F)F)ncn2O)=O)CC1C Cc1nc(CNC(=N)NCCOCCO)n[nH]1 N1(N2C(C3(O)CN(C(c4ccsn4)=O)C3)CCC2)CCCC12CCOC2=O c1(C(=O)NCCN(C(C2(CC=C)CC2)=O)C)cnn(C)c1CC C(=O)(CCCCCC(C)(C)C)Nc1cccc(NC(C2CC(C)=C(C)CC2)=O)c1 C1(NC(C(C)=CC2CC2)=O)CC2CCC(C1C)N2C(=O)CCC(=O)N(C)C c1(C(=O)NCC(C)NC(C2(C#N)CC(=O)C2)=O)cnc2c(c1)CCCC2 N1(C(CC2CC(=O)NC2=O)=O)CCCC(CC(=O)NCCC#N)C1 c1(C(N(CC(C)CNC(C2CCC(C)C2)=O)C)=O)cc(Br)n(C)n1 C1(CNC(C2(C(C)C)CC2)=O)CN(C(C2CCCS2(=O)=O)=O)CC(C)(C)C1 C1(NC(c2cn(C)nc2O)=O)CCC2(CC1)CN(C(C1CN(C3CCC3)C1)=O)C2 c1(C(=O)NCC(CCCC)NC(=O)CC2CN(C)C2)nc2ncccn2n1 Cc1c(C(=O)NCC2C(C)CCCN2C(=O)CCCc2ccsc2)c(Cl)nn1C C(C(=O)N=c1cc(C(F)F)[nH][nH]1)c1ccc(CC)nc1 C(CNC(C1C(C)C1C)=O)(CC(C)C)NC(CC(=O)NCC)=O c1(C(N2CC(C(C)NC(c3cncn3C)=O)C2)=O)cccc(=O)n1C N1(C(CC2(C(=O)OC)CC2)=O)CC(C(=O)NC2(C)CCCC2)C2(CCC2)C1 CC1CCC=C1C(=O)N1C2CCC1C(CNC(=O)CN1CC(=O)NC1=O)C2 N1(C(CC2(CC)CCC2)=O)C2CCCC1CN(C(c1ccoc1)=O)C2 C1(C2CCCC2)(NC(C(c2ccccc2)NC(C2CS(=O)(=O)C2)=O)=O)CC1 Cc1sc(NC(=O)CN2CCSC(C(C)C)C2)c(C)c1C C1(CNC(C2CCOC(CF)C2)=O)CC2(CC2)CN1C(c1ncc(C(F)F)s1)=O Cc1sc(Br)nc1C(N1CCCCC1C)C(=O)NCC1CCCO1 N1(C(C2(NC(c3ncnc(C)c3C)=O)CCN(C)C2)=O)CC2(CCC(=O)NC2)C1 CC1(C)CCCOC1CC1(CCC(=O)NC(C2COCCO2)=O)CCC1 N1(C(C=Cc2n(CC)ccn2)=O)CCN(C)C(CNC(=O)CN2CCCC2C)C1 C12(C(=O)NC3C(OC)C(C)(C)C3)COC(C1)C(NC(c1cc(C(C)C)on1)=O)C2 N1(C(C2N(C(c3cc(COC)on3)=O)CC(O)C2)=O)CC2CC2C1C#N c1(CNCc2c(C)nn(C)c2Br)cnc2ccsc2c1 c1(NC(c2ccc(F)cc2)CC)cc(Br)ccc1S(=O)(=O)NCC(C)(C)CC(F)F C1(C(N(C2CCSC2)C)=O)OC2CNCC1C2 C(=O)(CC(O)CNC(C)=O)NC1C(NC(Cc2c(CC)con2)=O)CCC1 CC(CCC(=O)NC(C)C(CO)NC(=O)CSCC(F)F)N(C)C C(=O)(N=c1cccn[nH]1)c1cccc(-c2ccc(-c3nccc(OC)c3)cc2)c1 C1(NC(c2c(CC)nc[nH]2)=O)CCSC12CN(C(=O)C=Cc1ccc(=N)[nH]c1)C2 c1(C(N(CCNC(=O)CC(F)(F)c2ccccc2)CC)=O)ccc2c(c1)COC2 c1(CCNc2cc(N(C3(NC(C)=O)CCC3)C)nc(C)n2)ccc(S(N)(=O)=O)s1 C1(C(=O)NC(C)CNC(c2c(Cl)nn(C)c2Cl)=O)CCn2cncc2C1 c1(C(N2C3C(NC(CSCCCC)=O)C(C3)C2)=O)ccnc(O)c1F C1(C2CC2)(NC(c2c(C)oc(SC(F)(F)F)n2)=O)CCOC1 CC(=O)CCCC(=O)N1CC(NC(C2CC2C2CC2)=O)CC(C)C1 c1(NC(CNC(c2cnn3c2CCCC3)=O)C2CCC2)nc2cccc(F)c2s1 c1(C(=O)NC(C2CCN(C(=O)C=Cc3ccc(F)cc3)C2)C)ccc(N)c(F)c1 C(=O)(C(C(C1CCC1)OC)N1CCC(CC(=O)OC)CC1)NC(CC)(C)C c12cn(nn1)CC1CN(C1)C(=O)N2.c1(CC2CCOCC2)nnnn1CC(F)F C(=O)(CN(C)C)N(C)CC1(CNC(C2CC2C(C)(C)C)=O)CC1 c1(OC)ccc(N)c(C(=O)N(CC(C)(C)NC(c2cncs2)=O)C)c1 c1(-n2c(C(=O)NCC(C)N(C(=O)C(O)C3CCCC3)C)ccn2)ccccc1Cl c1(C(=O)NC(C)CNC(c2cn(C)cn2)=O)cc2ccnc(Cl)c2[nH]1 C12(NC(C(c3ccc(Br)cc3)CC)=O)CCC(C1)N(C(=O)COCCF)C2 CN1C(=O)NCC1C(=O)NCC1(CNC(=O)COCC(F)(F)F)CC1 C1(C(=O)NCc2cn(CC3CCCC3c3ccccc3)nn2)CN2CCC1C2 C1(C)(C(=O)NCC(C)OCCO)CN(C(C2C3CC(=O)CC23)=O)C(C)(C)C1 c1(C(=O)NC2C(NC(C3(C#C)CCCC3)=O)CC2)ccc(C#C)c(F)c1 N1(C(C2C(=C)CC2)=O)CC(C2CCCCN(C(=O)Cc3cccc(Br)c3)C2)C1 C(C(CC(C)C)C(C(=O)Nc1ccc(F)cc1)N(C)C(C1CCC1)C)OC c1(OCC=C)c(C(=O)NCC=CCNC(=O)C=Cc2cn(C)nn2)cccc1C C(=O)(C(C)(C)CCCO)NCC1C(C)CN(C(C2CSCC(=O)N2)=O)C1 N1(C(C(C(=O)OC)OC)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)CC1C(F)F N1(C(c2ccnc(Br)c2F)=O)CC2(CCC(NCc3cnc(O)nc3O)C2)C1 N1(C(c2c(C)occ2)=O)CC(N(C)C(C2(n3cccn3)CC2)=O)C(O)C1 C(c1cccc2ccncc12)=Cc1cc(C(C)(C)C)no1 C#Cc1cccc(OCC(=O)NC2CN(C(=O)CCC(=C)C)C3CC23)c1 CC(CCc1ccccc1)CC(=O)NCc1cn(-c2ccn(C)n2)cn1 CCCC(C(=O)N1CCCC1C1(NC(c2csc(CC)n2)=O)CC1)S(N)(=O)=O C(=O)(C(C)(C)C(F)F)NCc1nccc(C(=O)NC(c2cn(C)cn2)C)c1 Cc1ncc(C(N2CC(NC(c3cc(C4CCC4)no3)=O)C(C)C2)=O)c(=N)[nH]1 C1(NC(C(C)Cn2cccn2)=O)COC2(CCN(C(=O)CCN(C)C)CC2)C1 N1(C(c2scc(COC)c2)=O)CC(C)OC2(CCN(c3cncc(C#N)n3)C2)C1 C1(NC(=O)C=CC2CC2)COC2(CCN(C(=O)COCC3CCCO3)CC2)C1 C1(NC(C2(COCC)CC2)=O)CC2C1CCN2C(c1cccc(C(F)(F)F)n1)=O C=CCC(C(=O)N(C(C)C(=O)NCC1CCCN1C)C)C(C)C C1(C(N(C)CCc2ccccc2)=O)CCC2(CC2)N1C(C1CC(C)(C)C1)=O c1(C(N(CCCN(C)C(c2ncn(C)n2)=O)C)=O)cc(Br)ccc1N c1(C(C(=O)NC(CCN(C(C=CCCC(C)C)=O)C)C)(F)F)cc(F)cc(F)c1 c1(C(N2CC(C(C(=O)NCC(C)C(F)(F)F)OC)C2)=O)ccnc(C)c1N CN1C(=O)NCC1C(N1CCCC1CCNC(c1ccc(C(C)(C)C)cc1)=O)=O Cc1cc(C(N2CCCC(O)(CCNC(C3CC3C)=O)C2)=O)c2cnn(C)c2n1 c1(C(C)C)noc2ncc(C(N3CCC(C)C3CNC(=O)C3=CCCC3)=O)cc12 C(CCC(C)C(=O)NCCCC(C)NC(C1CCCCC1(C)C)=O)OC Cc1nn(-c2ccc(F)cc2)cc1C(N1CC(CNC(=O)CO)C(C)C1)=O C1(C(=O)NC2C3CCN(C(C45CC(C)(C4)C5)=O)C3C2)CCCCN1S(=O)(=O)N(C)C C(=O)(C(C)(F)F)N(C1CCN(C(C2CC(CF)C2)=O)C1)CCC CC1CC(N(C)C(c2cc(CNC(=O)Cc3cn[nH]c3)cs2)=O)CCO1 c1(C(=O)NC(C(C)NC(C2C(C)CCO2)=O)(C)C)ccc(S(C)(=O)=O)o1 N1(C(CSC)=O)CCCC(O)(CNC(=O)CCC2(C)CC2)C1 N1(C(C=C(C)C(F)F)=O)CC2OCCN(C(=O)C(C)N3CC(C)C3)C2C1 C(=O)(C(COC)CC(C)C)NCC(CN(C(c1c(CC)nc(C)n1C)=O)C)C N1(C(C(C)CF)=O)CCC2(CCC2CNC(c2ncccc2N)=O)CC1 C12(NC(CC)=O)CCN(C(=O)CSc3nc[nH]n3)CCC1C2.c12cccc(c1)N2 N1(C(c2cc(OC)ncc2)=O)C2CCC(C2)C1C(=O)Nc1ccc(=N)[nH]c1 C1(C(=O)NC(CC=C)CC=C)CCC(C)(C)N(C(=O)C=C(C)C)C1 c1(OC)ccccc1C(=O)NCC(=O)NC1(NC(=O)CSC(F)(F)F)CCOC1 CC1(C)CN(C(=O)CC2CCCC(F)(F)C2)CC1NC(=O)CCOC1COC1 N1(C(C)Cc2ccccn2)CCC(NC(c2coc(CC3CC3)n2)=O)CC1C C1(CNC(C2(C(F)F)CC(=C)C2)=O)CCCCN1C(=O)C(C)Oc1ccccc1 N1(C(C(C(C)C)C)=O)CC2(CCOCC2)CC1CNC(=O)CC1CCCN(C)C1 C1(C(N2C(c3ccc(C)cc3)CCC2)=O)CC2(CC2)CN1Cc1c(C)n[nH]c1C c1(NC(=O)NCC2CC(=C3CNC3)C2)cc(Cl)c(Cl)s1 c1(OC)ccc(C)cc1NC(=O)C(CC1CC1)NC(=O)CC=C(Cl)Cl c1(C(=O)NC2CC(NC(CCCN(CCC)CCC)=O)C2)cc(Cl)c(F)cc1N N1(c2nc(SC3OCCN(C)C3)c3c(n2)ccs3)CCOc2ccc(F)cc2C1 CCC(CC(C)C)C(=O)N1CCOC(CN(C(=O)C(C)=C(C)CC)C)C1 c1(C(=O)NC2(CO)CCN(C(C3CCCS3(=O)=O)=O)CC2)cccc2nonc12 c1(C(=O)NCC(CNC(CCC(=O)OCC)=O)OC)nn(CC)cc1[N+](=O)[O-] C#CCC(CC(F)F)C(=O)NCC1CN(C(=O)C(C)SC)CC1c1ccccc1 C1(NC(c2cc(Cl)ns2)=O)C2CC3CN(C(=O)Cc4ccon4)C1C3C2 C1(CC2CC(CN(C)C)C2)CCOCC1.C12(CC1)C(=O)NN(C)C(=O)CO2 c1(C(=O)NCC(C2CC2)NC(c2nnn(C)n2)=O)cc2ccc(F)cc2s1 C1(OC)CCCCC1n1cc(CN)nn1.C12(CCOCC1)C(=O)N2 c1(C(=O)NCC(CNC(c2n(CC)ncn2)=O)C)c(C)cccc1[N+](=O)[O-] N1(C(C(C)(C)OCC)=O)CC2ON=C(CNC(c3ccc(F)c(F)c3)=O)C2C1 N1(C(CC(C(F)F)NC(C(COCC)N=[N+]=[N-])=O)=O)CCC(C)C(C)CC1 c1(C(=O)NC(CC(C)NC(CC2(COC)CC2)=O)C)c(C)cc(Cl)cc1C CC(C)CC(C)(C)C(=O)N1CCC(C)C(N(C(=O)COCC(F)F)C)C1 Cc1ccc(CC(=O)NC2CN(Cc3cc(F)ccc3Cl)CC2O)c(C)c1 c1(C(=O)NC(C)CNC(=O)CC2CSC2)c(O)nc(=O)n2c1CCC2 C1(CNC(c2c(CCN(C)C)cccc2)=O)CC2(CC2)CN1C(c1cc[nH]c1)=O CC(C)CC(C)CC(=O)NC(C)(C)CN(C)C(c1cnc(C(C)(C)C)[nH]1)=O C(=O)(CC(CC)C(C)C)NCC(C)(C)NC(Cc1c(SCC)cccc1)=O N1(C(COCC(OC)OCC)=O)CCOCC1C1(CO)CC1 c1(OC)cc(C(=O)NCCc2nc(C(F)(F)F)cs2)cc(OC)c1C(=O)NC C1(N(CC#C)C(C2(C)CC2)=O)CCN(C(C2CCC(=O)C2)=O)CC1 c1(OC)cc(F)c(NC(=O)CC2CCN(C(c3cnsn3)=O)C2)cn1 C1(S(N)(=O)=O)(C(N(CCOCCNC(C(C(C)C)OCC)=O)C)=O)CCCC1 C1(NC(c2cnc(C)s2)=O)CN(C(=O)C(c2c(C)n[nH]c2C)C)C2(CCCC2)C1 CC(C)(F)CCC(=O)NC(C)(CNC(c1cccnc1S)=O)C1CCC1 c1(C(=O)NC(CC)CNC(=O)CCN2CCCC2)cc2cc([N+](=O)[O-])ccc2[nH]1 N1(C(=O)CC2CCOC2)CC2CC(C1)N2C(=O)CC1CC(C2CC2)C1 c1(C(N2CC(O)(C(C)NC(C(CC)C)=O)C2)=O)[nH]c(C)c(C)c1C Cc1nn(C)c(C)c1C(=O)NCCNC(c1ccc(C(F)(F)C(F)(F)F)nc1)=O C12(F)CCC(CC1)CNC2=O.O=C(C(O)C1CC1)NCC1(O)CC1 C1(C(=O)NC(C(=O)N(CCOC(C)=O)C2CC2)C2(O)CCC2)CC(=O)OC1(C)C c1(C(=O)NC(C(C)NC(C2CCS2(=O)=O)=O)C)cc(F)cc2cnccc12 C1(NC(CN(C(=O)OC)CC)=O)CC(C)CN(CCc2ccccc2)C1 C12(NC(CCOCCOC)=O)CCN(C(c3cc(C4CC4)[nH]n3)=O)CC1C2 c1(C(C(=O)NCc2ccco2)N(CCCC=C)C)cn2cc(Br)ccc2n1.OCC C1(C(=O)NCCN(OC)C)CCN(C(C2CC2C2CCC2)=O)CCO1 C1(NC(C2OCC(C)C2)=O)CC(=O)N(C2CN(C(=O)CN(S(=O)(=O)CC)C)C2)C1 c1(SCC(=O)NCCN(C(c2coc(Br)c2)=O)CC)ccc(F)c(F)c1 C(=O)(CCCCC(=O)NC1CCCCC1NC(=O)C=CC1CCOC1)NC Cc1ccc(C(=O)C(=O)NC2(CO)CN(C(=O)C(C)(C)c3ccc(Cl)s3)C2)cc1 Cc1c(NC(c2cccnc2CO)=O)ccc(C#N)c1Cl.c12cccc(c1)NC2=O N1(C(C2C(OCC)CC2)=O)CCC(O)C1C(=O)NCc1ccn(C2CC2)n1 NS(=O)(=O)C(C(=O)NC1CC(NC(c2occc2C2CC2)=O)C1)c1ccccc1 n1(-c2noc(CN)n2)cc(Br)c(C)n1.C1(c2nnnn2C(C)(C)C)(SC)CCSC1 CN1CCCCC1CC(=O)NCC=C1CCN(C(c2cnns2)=O)CC1 c1(NC2CCCC(CO)C2)nc(=N)[nH]c(=NCC(CO)c2ccccc2F)[nH]1 c1(-n2cc(CC3N(C(c4c(C(=O)O)scc4)=O)CCC3)nn2)cccc(Br)c1 S(=O)(=O)(c1ccsn1)N1CC(c2n(C(C)C)ncc2)C1 C1(C(=O)NC2(C3CCCCO3)CC2)CCN(C(=O)c2ncccc2Cl)O1 C1(NC(C(C(C)C)NC(C2CCCC2F)=O)=O)CCC2(CC1)N=N2 c1(C2(C(N(C(C3CCCC(F)(F)C3)C(=O)OC)C)=O)CC2)c(F)cccc1Cl c1(CNCC2C(C(c3ncc(NC(CC(CC)C)=O)cn3)=O)C2)c(F)cccc1F C1(F)(C(=O)NCC2CCCC(NC(C(C(C)O)NC(C)=O)=O)C2)C(C)(C)C1(C)C Cc1cccc2c(C(N3CCN(C(c4c[nH]c(C#N)c4)=O)C(C)C3)=O)coc12 c1(C(=O)NC2CCCN(C(C(CC)n3nccc3C)=O)C2)cc(C#N)ccc1F C1(C(N2CCCC(OCCC)C2)=O)CCN(C(c2cc(C(C)C)sn2)=O)C1(C)C C1(CC(=O)NCC2OCCN(C(C3C(COC)C3)=O)C2)CCC(C(F)(F)F)N(C)C1 c1(C2C(C(=O)NCCCNC(=O)NC3OCCO3)C2)ccc(C(F)(F)F)cc1Cl c1(CC)[nH]nc(C(N2CC3CC2C3NC(=O)Cn2cccn2)=O)c1C c1(OC)cc2c(cc1C(N1CC3CCC1C(O)C3)C(=O)NC(C)C)OC(C)C2 CC1CCC(C)(C(N2CSCC2C(=O)N(CC(O)CO)C)=O)C1(C)C N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(C2CC2C(F)F)=O)C2CCCC12 N1(C(C(C)(C)OCCC)=O)CCCCC1c1cn(-c2cccnc2)nn1.C(C)=O C(CCNC(C1(S(N)(=O)=O)CC1)=O)(C(C)C)NC(C1(OC)CCOC1)=O N1(C(c2cc(OC)cc(C)n2)=O)CCC(C2CC(NC(C)=O)C2)CC1 N1(C(C(C)Nc2ccccc2[N+](=O)[O-])=O)CCc2nc(SC(F)F)nc(O)c2C1 C(C(C)(C)C(=O)NC1CN(C(C2CCS2(=O)=O)=O)C1)OC C=C(Cl)CCC(=O)N1CCOCC1CNC(=O)CCC1CC1(F)F N1(c2cc(C)ncn2)CCC(NC(c2csc(C3CCCO3)n2)=O)C(O)C1 CCC(CC(=O)NC1(C(=O)NCC2CC(F)(F)C2)CC(O)C1)C(C)C CC(C(=O)N1CCNC(=O)C1)(C(F)(F)F)n1nnc(-c2cc3c[nH]nc3s2)n1 C1(c2n(CC(=C)C)nnn2)(NCC2CCCCC2C)CCN(CC(F)(F)F)CC1 c1(C(=O)NCCCN(CCCNC(CCCC(C)C)=O)C)ccc2c(c1)OCC2 Cc1cc(C2CC2)ccc1C(=O)NCC(C)NC(=O)C(C)Cc1c(C)noc1C C(=O)(N=c1[nH]ncs1)NCc1ccccc1.N1(CC)CCC(CNCC)CC1 C1(NC(c2cn(C(C)C)nn2)=O)C=CCN(C(=O)C(c2ncccc2F)(F)F)C1 C(N=c1nc2sccc2c(N2CCOCC(C)(F)C2)[nH]1)c1nn(C)c(Br)n1 N1(C(C(C)OC)=O)CCN(C(C2CC3C=CC2CC3)=O)C(CCO)C1 N1(CC(=C)Cl)CCCC1C1CCCCN1C(c1nccc2ccccc12)=O c1(C(N2CC(NC(=O)CC3CCOCC3)CC(C)C2)=O)cnc2n1CCCCC2 C(=O)(CCCCSC)N1CC(CC(C(=O)NCCC(COC)OC)F)C1 C(=O)(C1CCc2nccn21)N1CC(=CCC)C1.C12CCC(O1)CNC2=O C(CC(C)C(=O)NCC1(C(=O)NC(Cc2ccco2)CO)CCCC1)=CCC N1(C(c2c(COC)onc2)=O)CCC12CN(C(c1cc3ncsc3[nH]1)=O)C2 C12(C(N3CC(NC(c4ccc(Cl)s4)=O)C3)=O)CCCC(CCC1)C2O C(=O)(C(C)CCCC(C)C)NC1CCN(C(c2cc(C)sn2)=O)CC1 Cc1ncc(Cl)c(C(=O)NC2CCCCC2NC(=O)C(C#N)C2CC2)n1 N1(C(CCCCCC)=O)CC2CCCN(C(=O)CCCc3ncc(C)o3)C2C1 c1(C(=O)NCC2(O)CN(C(C(C)c3ccco3)=O)C2)cncn(C)c1=O C=CC1CN(C(=O)C(C)(C2CC2)N(C)C(C2CCC(NC(C)=O)C2)=O)C1 N1(C(C2CC(CC)OCC2)=O)CCOC2(C1)CN(C(c1c[nH]c(=N)c(C)c1)=O)C2 c1(C(N2C(C)(CC(=O)NC3COCC3CO)CC2)=O)cccc2[nH]ncc12 N1(C(C(C(C)O)C)=O)CCN(C(c2ccccc2C(F)F)=O)CC12CCC2 CC(C)C(=O)C(=O)N1CCN(C2CN(C(=O)CC3(O)CCC3)C2)CC1 N1(C(C(N2CCN(CCN3CCOC3=O)CC2)=O)=O)CCC2(CC1)CC2 c1(NC(C(c2occ(C)c2)N(C)C(c2n[nH]c(C)n2)C)=O)cccc([N+](=O)[O-])c1 CC1(C)CC=C(C(=O)N2CC3CC(C2)CN(C(=O)Cn2nnc(=N)[nH]2)C3)CC1 c1(C(=O)NC2C(CNC(C=CCN(C)CC)=O)CCCC2)ccc(C)c(Br)c1 C1(NC(c2c(C)nc(O)cc2)=O)CN(C(=O)CC(C)(C)C(F)F)CC2(CC2)C1 c1(NC(C2N(Cc3c(OC)c(Cl)ccc3)CC2)=O)ccc2cn(C)nc2c1 C(=O)(C(C)(C)CCCNC(c1ccco1)=O)NCC1CCN(C(CC)=O)C1 c1(C(=O)NCC2CCC2C(N(C2CCS(=O)(=O)C2)C)=O)ccc(N)cn1 c1(OCOC)cccc(C(=O)NCCC(O)CNC(=O)C(C)N(C)C)c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC(CNC(C2CCCOC2)=O)C(O)C1 C1(CC#C)(C(=O)NCC(F)CNC(c2cnn(C)c2OC)=O)CCOCC1 C1(C(=O)NC(CN(C(c2nc(CC)sc2)=O)CC)C)CCCOC1CC(C)C c1(C(=O)OCC(C(CC)(C)C)=O)cc(Br)cc(S(C)(=O)=O)c1F C1(CNC(C(C)C2CC2)=O)CCCN(C(c2ccn(-c3ccncc3)n2)=O)C1 c1(C(=O)NCCC2CCN(C(C3C4CCC34)=O)C2)cncc(C2CCOCC2)c1 c1(OC)cc(NC(C2CCCN2C(C2CCCC2)=O)=O)ccc1C Cc1ccnc(NC(C2CCN(C(c3ccc(-n4ccnc4)cn3)=O)C2)C)n1 C1(C(=O)NCCCC(=C)Cl)(CNC(C2CC(=O)C2)=O)CC12CCC2 c1(C(N2C(CNC(CC3C(C)C3)=O)CCCC2)=O)cc2cc(N)ccc2[nH]1 c1(NC(CC(C)CNC(C2CC23CCOCC3)=O)=O)c(O)cccc1F Cc1nn(C2CCC2)cc1C(=O)NC1C=CCN(C(=O)C(F)(F)CO)C1 c1(C(=O)NC(C(C)NC(Cc2c(C)nc[nH]2)=O)C)cccc(CNC(C)=O)c1 CCCC(CCC)C(=O)NCC1CC(C)(C)CN1C(C1CCC1CF)=O c1(OC)cc(C)ccc1C(N1CCC(O)C(NC(C2(CN(C)C)CC2)=O)C1)=O c1(C(=O)NCC(C)(CNC(C2CC2Cl)=O)OC)ccc(CO)cc1C C1(C(N2C(CNC(C3CC3Br)=O)CC(OC)C2)=O)CCC2(CC1)CC2 C1(C(=O)NC2CC2)CCN(CC2(O)CN(C(CN(C(=O)OC)C)=O)C2)CC1 c1(OC)ccc2cnc(N3CCCC3C(=O)NCc3nc(Br)cn3C)nc2c1 Cn1ccc(C(=O)NCC2CN(C(=O)COCCF)C(C)(C)C2)cc1=O C(=O)(C(CCCC)C(C)C)NC1C(C(N(CCCC)CCO)=O)OCC1 CC(C)(C)CC(O)CC(=O)NCC1CCCN1C(=O)CSCC1CCCCO1 N1(C(CCSCC(C)C)=O)CCC(CCNC(=O)C(c2ccc(Cl)cc2)C)CC1 C1(C(=O)Nc2c(OC)cccc2)CN(C(=O)C(CO)OC)C(C)(C)C1 C1(NC(c2cc(C)[nH]n2)=O)CC2CC1N(C(c1cnc(C(C)C)o1)=O)C2 c1(C(=O)NC2C(N3CCC(OC)C3)CCC2)cc2occc2s1 CC(C)CCCC(=O)NCCN(CC(C)O)C(C12CC(C)C1C2)=O c1(C(N2CC(CNC(CC(=C)C)=O)OCCC2)=O)cc(F)c(Cl)cc1Cl c12ccc(s1)n(CC)c2=O.C1(C)CC(N(C)C)C1.C(C(N)=O)NC c1(OCC(=O)NC2C(NC(=O)CCCCCF)COC2)ccc(Cl)c([N+](=O)[O-])c1 C1(CNC(c2cscn2)=O)COCCN(c2nnnn2Cc2ccccc2)C1 C(=O)(C(F)C(C)(C)O)N1CCC(C(C)C)(C(N2CCC2CO)=O)C1 C1(S)CCCN(C(C)C(=O)NCC(C)(C)CNC(=O)C(C)O)C1.CC(=O)N N1(C(c2c(C(=O)OC)c[nH]n2)=O)CCC(O)(CNC(=O)Cc2cccc(O)c2)C1 c1(CN2CCCN(C(C3(C)C(C)(C(=O)OC)CC3)=O)CC2)ccc2c(O)n[nH]c2c1 Cc1cncc(CC(=O)NCC2CCN2C(=O)C(c2ccccc2)C2CC2)c1 C1(C=O)CC2(CCN(CC3CCN(N4C(C(C)C)CC4)CC3)C2)C1.C1CC1 N1(C(C(c2ccccc2)=O)=O)CCN(C(C2CS(=O)C2)=O)CC1CO C12(C(=O)Nc3ncccc3C3CC3(F)F)CC1CN(C(=O)COC(F)F)C2 c1(C(=O)NC2CN(C(c3c(C)snc3)=O)CC2F)cnc2ccccc2c1 Cc1ocnc1C(=O)NCC(Cc1ccccc1)N(C)C(c1ncn(C)n1)=O N1(CCOC)CCC(C(=O)Nc2cc(Br)ccc2OCC(F)(F)F)C(O)C1 C1(C(N(C)CCNC(c2nnn(-c3ccccc3)n2)=O)=O)COCC1(C)C CCCCC(C)C(=O)NC1(CCNC(C2CCN(C)C2=O)=O)CCC1 c1(CC)ccc2cc(C(N3CCC4(CCC4NC(=O)CC(F)F)CC3)=O)[nH]c2c1 c1(C(=O)NCC2C(NC(C3(CC=C)CC3)=O)COC2)cc2ccc(F)cc2o1 Cn1c(C(N2CCC(N(CCO)C(C3CCCS3)=O)C2)=O)cccc1=O N1(C(CCOCC)=O)CC2(CC(NC(C3CCC(Cn4ccnc4)O3)=O)CO2)C1 c1(OC)ccc(C(C(=O)O)NC(C2CCC2)=O)cc1 Cc1ccc(OCCC(=O)NC(C)C(CO)NC(c2cccs2)=O)c(C)c1 C1(C(=O)OCC)(CF)CCN(C(c2cn(Cc3cc(CO)on3)nn2)=O)C1 CCCC(C(=O)N(C)CC1CN(C(=O)CCC(F)F)CCO1)C(C)C CCC(C(=O)N1CCCC1Cn1cc(C(=O)NCCOC(C)=O)cn1)n1cccn1 c1(OC(C(=O)NC2C(NC(CC=CCC)=O)CCC2)C)ccc(OC)cc1 C(CCC(C)CC(=O)N1CCC(NC(c2n[nH]c(C)c2Cl)=O)CC1)=C(C)C CCC(C(=O)NC1CC(C(N2CC3(C)CN(C)CC3(C)C2)=O)C1)C(C)(C)CC N1(C(c2cc(C)n(C)c2C)=O)CC2(CCC2)CC1C(=O)NCCC(O)C(F)F c1(C(=O)NCC2CC(NC(=O)CCCn3ccnn3)C2)ccc2c(c1)NC(=O)C2 C1(NC(=O)NC(COCC)(C)C)CCCN(n2nccn2)C1 N1(C(CC=C)=O)CCCC2(NC(=O)Cc3cccc4c(C)csc34)CCCC12 c1(C(=O)NC(C)Cc2csc(CNC(=O)CCCF)n2)cc(O)c2sccc2c1 CC1(C)CC(CC(N2CCOC3CC23)=O)N(C(=O)C(CO)NC(N)=O)C1 C1(c2n(CCSC)nnn2)(NCC(CC(C)C)C(N)=O)CC2(CCC(C)(C)CC2)C1 Cc1cc(I)c(F)cc1NC(=O)Cc1cc(=O)cc[nH]1 c1(C(N(C)CCNC(C2(F)CCCC2)=O)=O)ncn2c1CCC2 N1(C(CC(C(C)C)O)=O)CC(CNC(=O)Cc2nncn2C)OC(C)(C)C1 c1(NC(c2c(-c3c(OC)nccn3)ncs2)=O)cc(C)c(I)c(C)c1 c1(C(=O)NCC(CC)NC(c2nn[nH]c2C2CC2)=O)c[nH]c(=NC)s1 n1(CC)c(N(c2cnc(NC(C)=O)nc2)C)nnc1C1C=CCCC1 C(C)(C(=O)NC1CC(NC(=O)C(N2CCC(C)CC2)=O)C(O)C1)(C(C)C)OC c1(C(=O)NC(C)C=CC(=O)NCC(C)(O)C2CC2)cc(OC(C)(C)C)cc(=O)o1 Cc1cccc(F)c1CC(=O)NCCCCCCN(C)C(C1CCCN(C)C1)=O C1(NC(Cc2cnc(C)[nH]2)=O)CC2CC(NC(C3CNC(=O)C3)=O)C1C2 CC1(C)CCC(CNC(C2CC2CNC(C2COC2)=O)=O)OC1 C1(C(N(CCOc2ccc(C)cc2Br)C)=O)CN(C(=O)C2CC2)CCC12CCC2 n1(CC(=O)NCC2CCCN(C(C(CC)C#N)=O)C2)cc2ccccc2n1 c1(NC(CC2CCN(c3ccc(C(N)=O)cn3)C2)=O)c(F)ccnc1Cl c1(CNC(CCOCC)=O)cc(C(=O)NCc2cncn2C)n(C)n1 CC1(C)COC(CCC(=O)NC2(CNC(=O)Cc3sccc3Cl)CCOC2)C1 C1(N(CCO)Cc2[nH]nc(CC)n2)CCN(C(=O)CC2CC2)CC1 C#Cc1cncc(C(=O)N(C2(C(N3CCN(C)C(CC)C3)=O)CCC2)C2CC2)c1 c1(C(=O)NCC(C)N(C(=O)C(F)C2CC2)C)cc(F)cc2ccoc12 N1(C(c2c(C)nsc2C)=O)CC(C)C(C)(C(=O)NCC2CC23CCOCC3)C1 C=CC(F)(F)C(=O)N1CC(O)(CCNC(c2ncccc2C2CC2)=O)C1 C=CCC(CC(C)C)C(=O)NCCC1(C(=O)NCC2(CSC)CCCCC2)CC1 CC(C)(C)C(CNC(c1ccsc1C#N)=O)C(=O)N1CC(CO)C1 C#CCC1C(=O)N1.C(CO)(C(C)CC)NC(=O)CSCCC C1(F)(C(=O)NCC2N(C(=O)CCn3ccnn3)CCC2)CC2(CCC2)C1 C(N=C(NC1CC1)N1CCN(c2ncccn2)CC1)C1C(C(N)=O)C1 C#CCC(C(=O)N1CCC(CC)(CC)C1)NC(c1cc(C(C)C)[nH]n1)=O c1(C(=O)NCC2CN(C(C3C(C(C)(F)F)C3)=O)CC2(C)C)coc2cc(O)ccc12 C1(C(C)CNC(=O)Cn2nnc(=O)[nH]2)CCN(C(=O)C=CCF)CC1 N1(C(CC2(COC)CC2)=O)CCC(CO)C(NC(c2oncc2C)=O)C1 c1(CNC(C2(NC(N)=O)CC2)=O)cn(CC2CCCOC2)nn1 C=CCC(CC)C(=O)NCC(=C1CN(C(C2(C(C)C)CCC2)=O)C1)F c1(NC(C)=O)cnc(C)c(C(N2CC(CCNC(c3ccn(C)n3)=O)C2)=O)c1 N1(C(c2ccc(C)nc2N)=O)CCC2(CCC2)C(NC(C2CCN(C)C2=O)=O)C1 C1(C(N2CC(CN(C(CC(C)c3ccccc3)=O)C)C2)=O)CC(=O)N(C2CC2)C1 C1(NC(c2cncc(O)c2)=O)CCC(O)CN(C(=O)CC2CCCCCCC2)C1 C(=O)(C(C)(C)CCCNC(c1c[nH]c(Br)c1)=O)Nc1cn(CC)nc1 CC(C)C(F)(CNC(C1CC(F)(CF)C1)=O)C(=O)NC12CCN(CC1)C2 c1(C(c2n(CC(=C)C)nnn2)NCc2cc(O)nc(S)n2)ccc(C)c(Br)c1O CCCC(CCCNC(=O)CCCc1nncn1C)NC(C1(CO)CC1)=O N1(C(C(c2nn(C)c(CO)c2)=O)=O)CC(C2CN(C(=O)CC3(C)CC3(Cl)Cl)C2)C1 C(=O)(CCCC(N)=O)NC(C1(O)CN(c2cc(C(F)(F)F)ncn2)C1)C C(=O)(N1CCCc2nccn21)C1CC(O)CCN1Cc1ccc(C(N)=O)o1 CCCC(CC)C(=O)NC(CNC(c1c(F)cccc1Cl)=O)C1CC1 c1(C(N2CC3CCN(C(c4c(C)nsc4)=O)C3C2)=O)ccc2c(=N)[nH][nH]c2c1 c1(C(N2CCC(CNC(c3c(C(C)C)ocn3)=O)C2)=O)cnn2ccn(C)c12 C(=O)(C(C)CS(C)(=O)=O)NCC(CCCC)NC(=O)C(CC)CC C1(CN(C(=O)CCc2nc(C)cs2)CC)CCCCN1C(C1CCCNC1=O)=O N1(C(Cc2ccn(C)n2)=O)CCN(C(=O)NC23CC(CO2)C3)CC1 c1(NC(C(=O)NCCCC#CC)=O)ccc(Br)cc1C N1(C(C2CN(C)C2)=O)CC=CC(NC(C2CC(=O)N(c3nccs3)C2)=O)C1 C1(C(=O)NCCc2cccc(C(=O)NC)c2)CCC(=O)N(CC(F)(F)F)C1 Cc1ccc(C(=O)NCCCC(C)NC(C23CCCC2(C(N)=O)C3)=O)nc1C O=C(C#CC1CCC1)NCCCN(C(=O)CCc1ccc(Cl)nc1)CCO C12(CCCCC1)CC(=O)N1CC(O)(C1)CNC(=O)C2.c1(CN(C)C)cccn1C N1(C(=O)OC(C)(C)C)CCC2C(F)(F)C12C(=O)OCc1ncc(Br)cc1C#N.SC Cc1ccc(C(F)(F)F)cc1CC(=O)NC1CCC(NC(=O)CCN(C)C)C1 N1(C(c2nnc(C(C)(C)C)s2)=O)CCCCC(NC(c2cccc(O)c2F)=O)C1 C1(C(=O)NC2(CC=C)CCCC2)CN(C)CCN1C(C1OCCCC1(C)C)=O c1(C2(C(N3CC(n4cc(CC(C)(C)O)nn4)C3)=O)CCCC2)cccc(C#N)c1 c1(N2CC(CC)(CO)C2)[nH]c(=NC2COC(c3ccccc3)C2)nc2sccc12 C1(C(=O)NCCC2CC(NC(COC)=O)C2)CCOC(=O)CC1 C1(CN(C)C(C2CCC(C(F)(F)F)CC2)=O)CCCN(C(c2cncn2C)=O)C1 C1(C(=O)N(C(C)C(C)C)C)(CC)CCCN1C(C1CC1C1CC1)=O c1(C(c2cn(CC(C)NC(c3ccc(CC)s3)=O)nn2)O)ccc(F)cc1 C1(NC(CCC(=C)C)=O)CN(C(=O)Cc2ncc(C)s2)C(C)(COC)C1 N1(C(CC=CCNC(c2cc[n+]([O-])cc2)=O)=O)CCCC2(C1)N=N2 c1(C(=O)NC2C=CC(C(=O)NCc3cn(CC#C)nc3)C2)cnc(O)c(F)c1 N1(C(CCC(C)c2ccccc2)=O)CCC(C)C(NC(C2(S(N)(=O)=O)CCC2)=O)C1 N1(CC(CC)OC)CCC2(CC1)CN(C(c1cnn3cccnc13)=O)C2 C1(C(N(CCC#C)C)=O)CCC(NC(=O)C(C2CC2)OCC)CC1 C1(NC(CSc2n(C)ccn2)=O)CCCC(NC(c2cc(C(N)=O)cs2)=O)CC1 c1(C(=O)NCC(CNC(=O)CNC(=O)CCCCO)O)nc(Cl)ccc1F N1(C(COCCC)=O)CC2(CCC(NC(c3cc(F)cc(Cl)c3)=O)CC2)C1 C1(NC(CCSC)=O)CC1C1CCN(C(=O)C(N2CCCCCC2)C)CC1 c1(CC(=O)NCC2C(NC(CNC(C(CC)CC)=O)=O)C2)c(O)ncnc1O C=C(C)CCC(C)CC.c1(C(=O)N)cc(CNC(=O)C(C)n2cccc2)[nH]n1 c1(C(=O)NC(C)(CNC(c2ccoc2)=O)CO)ccc(Cl)c2c1OCCO2 C1(CNC(c2c(C)coc2)=O)CC(C)N(C(=O)Cn2ncc(Br)c2C)C1 Cc1cc(CO)c(SC2CCS(=O)(=O)CC2)cc1F c1(C(=O)NCC2N(C(CSC)=O)CC(O)C2)ccc(SC(C)=O)c(C)c1 C1(C(N2CCC(NC(C(C3CCCOC3)OC)=O)C(F)C2)=O)CC2(CCCC2)CO1 C1(C(N2CC(OCCC(=O)N(C)CC3CCOC3C3CC3)C2)=O)CCCCC1(C)C N12CC(CC1=O)C(=O)N1CC2C1.C(=O)(C=CS(C)=O)CN(CC)CC1CCCC1 C1(NC(COCC)=O)CCC2(CCCN2C(c2ccc(CNC(=O)OC)o2)=O)CC1 C1(CN(C(=O)Cc2ccon2)C)CCCC(NC(c2cncnc2)=O)C1 CC1(F)CCCCN(C(C2CC(O)CCN2Cc2ncc(Cl)nc2Cl)=O)C1 Cc1noc(C)c1C=CC(=O)N(C1CCN(C(C2CC3CC3C2)=O)C1)C c1(CCC)ccc(C(=O)NCC2CC2NC(C2(C(F)(F)F)CC2C(C)C)=O)o1 C=C=CC(C)C(=O)NC1CC(CCC(=O)NCc2nccc(C)n2)C1 C1(CC(=O)NC2(CNC(C3CC(n4ccnc4)C3)=O)CCCC2)CCCCO1 c1(CNCc2c(C)csc2)ccc(-c2cnc(=N)[nH]c2)cn1 N1(C(c2c(C)c(CO)ccc2)=O)CCC2CN(C(=O)C(C)n3cccn3)C2C1 c1(OCC)cnc(C(N2CCC(CNC(c3ncc(Cl)n3C)=O)CC2)=O)cn1 C#CCC(O)C(=O)NCC1CCN1C(c1c(-c2ccccc2)noc1C(C)C)=O N1(CC(C)(C)C(=O)NC2CCN(C(C3CC(O)CN3)=O)CC2)CCC(C#N)CC1 c1(NCC2(COC)CCCO2)[nH]c(=NCC2(S(C)(=O)=O)CCCC2)nc2scnc12 c1(NC2C(c3ccn(CCOC)n3)OCC2)nccc(=NC2CCC(C)(C)C2)[nH]1 C1(C(=O)NC2CC(CNC(c3cccc(NC)n3)=O)C2)CNC(=O)CC12CCC2 C(CC(C(=O)N1CCC(O)(CO)C1)NC(=O)C(C)C(F)F)=CC N1(C(CC)CC)CC(C(N2CC(C(C)NC(=O)COCCCOC)C2)=O)CC1=O CC(C)CCCC(=O)NC1(C(N2CC(C#N)(CCF)C2)=O)CSC1 CCCCCCC(=O)N1CCCC(C(=O)NC(C)(CO)C2CC2)CC1 c1(C(=O)NCC2C(NC(=O)CC3COCCO3)CC2)ccn2ncc(CO)c2n1 n1(CCC=C)c(N2CC(F)CC(F)C2)nnc1C1CCCc2ccccc21 N1(C(c2cccc(C)c2F)=O)C2CCC1CC(N(C)C(C1CC3CC1C3)=O)C2 CCC(CCC(=O)NC1CCN(C(=O)CCSc2nnnn2C)CC1O)OC C(C(C)(C)CN(C(=O)CC1CCN(C(=O)C(c2cnn(C)c2)O)C1)C)OC C(C)(CSC)(C(=O)Nn1cnnc1C)NC(CCC=C=C)=O C1(C(C)C)CCC(C(=O)NCC2(n3ccnn3)CC2)N1C(=O)C(O)CCN(C)C Cc1cnnc(C(N2CC(O)(CNC(=O)CCOCCN(C)C)C2)=O)c1 Cn1nc(C(=O)NC2CCCN(C(=O)CCCN3CCCCC3)C2)cc1C1CC1 N1(C(C(C)CC(F)F)=O)CCC2(C)CN(C(C3CCOC(=O)CC3)=O)CC12 N1(CCCCCNC(COCCCCCC)=O)CCCC(C(N)=O)C1 n1(CC)c(C)nn(CC(=O)NCCC(C)N(C)C(C2(C)COC(=O)OC2)=O)c1=O C(CCN(CC(C)C)N1CCC2(CCCN2C)C1)OC c1(C(=O)OC)ccc(N)c(C(=O)N(CC(C)NC(C2(CF)CC2(F)F)=O)C)c1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCCC(NC(=O)C(F)(F)c3cncs3)C2C1 C1(NC(=O)C2=COCCC2)CC2(CCN(C(=O)Cc3ccccc3O)C2)C1 N#Cc1cccc(CNC2CC(NC(=O)C=Cc3ccc(O)cc3)C2)c1 Cc1cc(-n2cc(-c3cnn(C)c3CNC(c3ccc(F)s3)=O)nn2)cc(F)c1 c1(C(=O)NC(CCCCNC(CC2(OC)CC2)=O)C)ccc(F)cc1Cl N1(C(CCCCC=C)=O)CCCCC2(CCN(C(=O)C(C)COC(C)=O)C2)C1 S(=O)(=O)(c1ccc(CNC2(C(=O)O)CN(C(C)=O)C2)c(Cl)c1)NCC(=O)OCC c1(C(=O)NC2CCCN(c3nc(C#N)cc(C)n3)C2)cccc2ccncc12 c1(CC(=O)NC(C(=O)NCC=C(Cl)Cl)C2CCC2)cccnc1F CC(N=c1ccnc(NCc2cccc(N3CCCC3=O)c2)[nH]1)C1CCOCC1 c1(OC)ccc(C(N2CCOC(CN(C(=O)CC3CC(C)=NO3)C)C2)=O)nc1 C1(NC(c2cc(CCC)ncc2)=O)C2CCN(C(=O)Cn3ccnc3C)CC12 C1(NCCOCC(C)C)CCCC1(C)N(C)C(C)C c1(NC(C2C(C)N(C)CCC2)=O)cc(C(C)(C)C)n2ncnc2n1 C1(O)CCCCCC1.C(=O)(CCN(C)C)N(C1CCC1)C(C)C Cc1[nH]nc(C(=O)NC2(C)CCN(C(=O)CC3CCC(C)(C)O3)C2)c1Cl Cn1ncc(C(=O)NCCCCC2CN(C(c3cnc(C(F)F)s3)=O)C2)n1 N1(C(c2nccn2C(C)Cc2ccccc2)C(=O)NC)CCOCC(C(=O)OC)C1 CC1CN(C(C2(F)CCCOC2)=O)CC1NC(c1nccn1C)=O N1(C(=O)Cn2cnnn2)CCC(NC(C23CC(C2)C3)=O)C(CO)CC1 C1(C(N2C(C(=O)OC)C=CCC2)=O)CN(C(c2nn(C)cc2C)=O)CC1(F)F C(C(F)(F)C(=O)NC1CC(C)N(C(=O)CSCCC(C)C)C1)OC Nc1cccc(C(=O)NCc2cn(C3CCN(C(=O)CN4CCC4C)CC3)nn2)c1 C1(NC(C(CC)OC)=O)CCN(c2nc(C(=O)OC)cc(C)n2)CCC1CO C(c1cccs1)=CC(=O)NCC1(C(=O)NC2CN(CC(F)F)C2)CC1 C(C(C)(C)C(=O)NCC1CC(C)N(C(=O)CCc2ncc(F)cn2)C1)OC c1(C(N2CCCC(O)(CNC(CCC(C)(C)F)=O)C2)=O)cccn2cncc12 C1(CNC(C(CC)C)=O)(OC)CCN(C(C2(OC)CC(CF)C2)=O)CC1 N1(C(=O)NC(C)CN2CCCC(C)C2)CCc2c(ccn(C)c2=O)C1 C(=O)(C#CC1CCOC1)NCCN(C(c1cc(C(C)(C)C)[nH]c1C)=O)CC C1(C(C)C)C(C(=O)NCC2CCC(=O)NC2)CCN1C(c1nccs1)=O C(=O)(CCCCCNC(=O)COC)NCCC1CN(C(C=CCC)=O)CC1C N1(C(N(CC=C)OC)=O)CC(C2(c3nn[nH]n3)CC2)C1 c1(C(=O)N(CC2CC(NC(=O)COCC3CCCO3)C2)CCO)cnc(Br)o1 Cc1ncccc1C=CC(N1CCC1CNC(=O)CC(O)C1CCCC1)=O C(=O)(CC(C)(O)CCC)NCC(=C)CCNC(c1ccc(OCCOC)nc1)=O CN=S(C)(=O)c1ccc(C(=O)N(C(C)CNC(=O)CCn2ccnc2)C)cc1 Cc1ccc([N+](=O)[O-])cc1C(N1CC(NC(=O)C(C)C(C)O)CC1C)=O N1(C(c2ccc(C(F)F)o2)C(=O)NC(CC)C)CCOCC(O)C1 c1(Nc2cc(C(=O)OC)no2)cc2c(s1)CCN(C(=O)C(C)(C)OC)C2 c1(CNC(=NCC)NCc2cnc(-c3ccccc3)o2)ccc(C)c(C#N)c1 C1(NC(C=C(CC)C)=O)CC2(C1)CN(C(C1(c3ccc(Br)s3)CC1)=O)C2 CC1=C(C(=O)NCC(F)CNC(C2CCCCN2C)=O)C(C)(C)CCC1 c1(C(=O)NC2CCC(CNC(c3csnc3Cl)=O)C2)ccc(=O)n(C2CC2)c1 C12(C(=O)NC3C4(CC(NC(c5cnc(O)s5)=O)C4)C3)CC3CC(CC1C3)C2 c1(C(C(=O)C2=COCCO2)=O)cnc2ccnn2c1.C(CCCC1CNC1)N C1(CNC(CCCC=C)c2nnnn2CC2CCOCC2)CCC(C)(C)CC1 C1(CC(N2CCC(O)(CN(C(=O)C(C)(C)CF)C)C2)=O)CCC(C)(O)CC1 c1(C(C)(C)NC(=O)OCc2cnc(C3CCC3)s2)ccc(C(F)(F)F)cc1 N1(C(c2c(SC)ccs2)=O)CCCC(NC(=O)CCc2cccnc2F)C1C c1(C(=O)NC2CC(n3cc(C(CC)(O)CC)nn3)C2)cnc2c(c1)COCC2 c1(CN(C(c2c(C#C)c[nH]n2)=O)CCN2CCC(O)CC2)ccc2ccoc2c1 N1(C(C2(C(=O)OC)CC2)=O)CCCCC(CNC(C2(C)CC3CCC2O3)=O)C1 c1(OC)ccc([N+](=O)[O-])c(NC(=O)NCC2CC23CCc2ccccc23)n1 C1(CNC(=O)CC2CC3(CCC3)CO2)CCC2CN(C(=O)Cc3ccsc3)CC12 C(=O)(C(C)CC(C)(C)C)NC1C(F)CCN(C(CCOCCN(C)C)=O)C1 c1(C(=O)NC2CN(C(C3CCC(C)(C)CO3)=O)CC2O)ccc2c(c1)CNC2=O Cc1nc[nH]c(=NCc2ccccc2CNC(=O)C(F)CC2CCCCC2)c1F Cc1scc(C(=O)NC(C(=O)NCC(c2nncn2C)C)C2CCCC2)c1C Cc1cc(Cl)ccc1OCC(=O)NC1CN(C(=O)CC2COC(C)(C)C2)C1 CC1(C)CC(CNC2CC3C=CC2C3)CCO1 c1(C(=O)OC)cnc(C(=O)NCC(C2CC2)NC(=O)C(O)C2CCCC2)cn1 C1(OC(C(C)N(CCn2ccc(C)n2)C(=O)OC)=O)COc2ccccc2O1.OCO C(=O)(CS(F)(F)(F)(F)F)N(CCCNC(C(CCCC)C)=O)C c1(CCC(=O)NCC(C2CCN(C(=O)CCOC3CC3)CC2)F)ccccc1Cl c1(C(=O)NC2CC2CNC(C2CCCCC2C(=O)N)=O)cccnc1O.C1(S)CC1 Cc1cn2cc(C(=O)NCCC(C)N(C)C(C3CCC3(F)F)=O)cc(F)c2n1 C12(CNC(N(CC(C)(C)C)Cc3ccc(Br)cc3)=O)COCCN1CCOC2 c1(CC)n[nH]cc1CNC(=O)C(C)=CCNC(C1CCC1C(=O)OC)=O C(=O)(C#CC1(C)CCCO1)N(C1(Cc2ccc(OCC)cc2)CCC1)C1CC1 c1(CC)cc(C(=O)NC2CC(C)(CNC(=O)C(C)CSC)C2)oc1CC N1(C(COC(CC)(C)C)=O)CC2CC(O)C1C2NC(=O)CCn1cc(C)cn1 CCN=C(NCc1cncs1)NC(C)CCS(C)(=O)=O c1(C(=O)NCC2(N(C(=O)CCc3ccc[nH]3)C)CC2)cc(C2CC2)cc(Cl)c1 C1(C(=O)Nc2c(C)cnn2C)COC2(C1)CN(C(=O)CCCCNC(N)=O)C2 c1(NCCSC)ccc(C(C(=O)OC)C=C(C)C)cc1 c1(CNC(C=CCN(C(CCSCCCC)=O)C)=O)nc(C)c(C)s1.NCC CC(=O)CCCC(=O)NC1CCC(NC(C2C(C)C2(F)F)=O)CC1 C1(C(=O)OCC23CC(C)(C2)OC3(C)C)CCc2ncc(Br)n2C1 C(=O)(C(C)(C)CC(=O)NCC1(CNC(C2CC3(CSC3)C2)=O)CC12CCC2)OC Cc1nnc2cnc(C(N3CC(CNC(c4cscn4)=O)OC(C)(C)C3)=O)cn12 c1(C(=O)OC)ccc(NC(C2C=CCN2Cc2ccnc(Br)c2F)=O)c(Cl)n1 C1(C(N(CCN(C(=O)CC2CCCNC(=O)C2)CC)CC)=O)CCCC1C1CC1 C1(CCC)(NC(=O)C(COC)NC(=O)CN)CCN(C(C2CC2(Cl)Cl)=O)CC1 N1(C(N2CC(OC)C(F)(F)C2)=O)CC(C)Oc2ccncc21 C[Si](C)(C)C1CCCC(C(N2CC(c3cn(CCCNC=O)nn3)C2)=O)C1 C(=O)(CC(C)CC(C)(C)C)NCN1CC2CCN(C(c3cc(C)[nH]c3C)=O)C2C1 c1(C(=O)NCC2(F)CC(NC(c3cc(C)oc3)=O)C2)nc(C(C)C)oc1C CCC(CC(F)(F)F)C(=O)N1CCOC(CNC(=O)CCC2CCCO2)C1 N1(C(c2c(C)nsc2C)=O)CCC(C2CCCN(C(=O)CN3CCCC3=O)C2)C1 N1(C(C2C(C(=O)OCC)C2)=O)CCC2CCCC12C(N1CCC(n2cnnn2)C1)=O c1(-n2cc(C3CN(C(C(COC)(C)O)=O)C3)nn2)ncnc2ccsc12 c1(C(=O)OC(C)(C)C)cc(C(=O)O)c2ccccn12.N12CCCCC1C2C C1(C(N(C2CCNCC2)C)=O)CCCN(CC2CCCC2(C)C)C1 N1(C(Cc2cc(C)no2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CC1C1CC1 Cc1cnc(C(=O)NC(c2cn(-c3cc(F)ccc3F)nn2)C)cc1C c1(OC)ccc(Br)c(CNC2CC(C)CN(C(C34CCC(CC3)CC4)=O)C2)c1 S(=O)(=O)(c1ccc(N(C)CCN(C)C)c(Br)c1)NCC1(C)CCC(C)CC1 C1(NC(C(C)OCCOCC)=O)CCN(C(=O)CC2CC=CCN2C)CC1 Cc1nc(O)ccc1C(=O)NC1CN(C(c2cnc(O)c(F)c2)=O)CCC1C c1(C(=O)NC2CCC(SC)C2)ccc2ncsc2c1 C1(CC=C)(NC(c2cnn(CCO)c2)=O)CCN(C(=O)C(C(C)C)N(C)C)CC1 Cc1cc(C(=O)NOCC(=O)NCC(C)CC(C)C)[nH]c1C CCCCC(C)(F)C(=O)N1CC(CCCCNC(c2cn3nc(C)sc3n2)=O)C1 C#Cc1cnc(C(N2CCOC(CCCNC(c3c[nH]nc3Cl)=O)C2)=O)c(C)c1 Cc1ccc(C(=O)NCC(C)CN(C)C(C2(C)CCC(C)C2)=O)c(C)n1 Cc1nnc(C(=O)N(C(CNC(=O)CCC2CC2)C2CC2)C)o1 Cc1cc2sc(C(=O)NCC3CCC3NC(c3sccc3C)=O)c(C)c2cc1C CC1CCCCC1(CNC(c1ccc(O)cc1F)=O)NC(c1cnn2c1CCC2)=O c1(NC(CC#CC)C)ccc(S(=O)(=O)NCc2c(C)noc2C)c(Br)c1 c1(C(C(=O)NCCCNC(=O)CC2CC2(F)F)O)ccc(Cl)cc1F CC(N=c1ccnc(N(C)Cc2ccn(C)n2)[nH]1)c1ncc(F)cc1F C1(NC(=O)OC)N(C(=O)CCNC(=O)CN(C)C(=O)C2CC2)CC1(C)C Cc1cc(C(N2CCC(N(C(=O)CCOC(C)C)CCO)C2)=O)c(C)s1 CCC(C)(O)C(=O)N1CCC(C(C)NC(c2cccc(OC(C)C)c2)=O)CC1 N1(C(C(C)Cc2ccccc2)=O)CC(NC(C2CCC(=O)N2C)=O)C(F)C1 c1(OC(C)C)ccccc1C(N1CC2CC1C2NC(=O)C(=O)NC1CC1)=O c1(CN2C(C)(C(=O)Nc3cc(C)c(Br)cn3)CCC2)ccc2nonc2c1 c1(OC)ccc(NC(C2CC3(C2)CN(C(=O)CCN(C)C)C3)=O)cc1Br c1(C(=O)NC(C2CN(C(=O)C3=NNC(=O)CC3)CCO2)C)ccc(Cl)c(F)c1O Cc1ncc(C(=O)Nc2cccc(NC(=O)CCC3CCC(=O)NC3)c2)cc1N c1(C(=O)NCCC(C)NC(=O)CC2CCC(C)(C)C2)cncc(-c2ccoc2)c1 C(C(O)CCCO)NC(c1cc(CNC(C2CCCOCC2)=O)[nH]n1)=O C1(CCC)(NC(C2CC2Cl)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1 Cc1cc(F)c2c(c1)CCN(C(c1ccc3c(c1)OCC3)=O)C2 C1(C(N(CCOC)C)=O)CC2(CCN1C(=O)Cc1cnccc1C)CC2 CCC(C)(C(=O)N(CCCNC(c1csc(-c2cccc(Cl)c2)n1)=O)CC)OC c1(CNC(C2C(C(N3C(C)COCCC3)=O)C2)=O)c(F)ccc(F)c1Cl N1(C(C(c2cncnc2)C)=O)CC2(CCC2)CC1C(=O)NC1COC(C(F)F)C1 CC(CC(F)F)C(=O)NCCOCCC(=O)NCCc1c[nH]nc1C1CCCO1 CCC(C)(CNC(C1(F)CCCN(C(c2cc(OC)ns2)=O)C1)=O)C(N)=O c1(OC)cnccc1CN=C(NCC(=O)NC)NC1CCC1 C(=O)(C(F)(CNC(C1CC1C1CC1)=O)C(C)C)NCC1(C#C)CCOCC1 c1(NCCC(CC)O)nc(N2CC3COCC(C3)C2)nc2c1ncn2C(C)C C12(NC(CCC)=O)CCN(C(=O)Cn3ccnc3C=CC(=O)OC)CCC1C2 C1(CC)CN(C(c2nocc2C)=O)CCC1NC(=O)CNC(C1CCCC1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(C)CCC(CNC(=O)Cc2cccnc2O)C1 C1(NC(CC=C)=O)CN(C(c2ccc(Br)c(OC(F)(F)F)c2)=O)CCC1(F)F c1(C(=O)NC2C=CC(CC(=O)NCC(C(CC)C)C)C2)cccc(C)c1N c1(CNC(=O)NC2CCCC2CNc2ccccc2)ccc(F)cc1C1CC1 C(=O)(C(O)CNC(=O)C=C(C)C)NC(CC)COC(C)C C(=O)(CCC1CCc2ccccc21)NCC(CNC(C#CC1(C)CC1)=O)(C)O c1(NC2CCN(C(=O)NCC#CC)C2CCC(C)C)cccc2c1CCCC2 CC(C)(C)CCC(=O)C(=O)N1CCC(C)(NC(c2cc3ncccn3n2)=O)CC1 c1(CC(=C)C(=O)NC(C)CCCN(C)C)ccc(F)cc1F N1(C(c2cc(C)oc2)=O)CC2(C1)SCCC2NC(=O)C(O)C1=CCCCC1 c1(-c2n(C(C)C(F)(F)F)nc(-c3cncc(Br)c3)n2)ccc(Cl)cc1Cl N=c1sccn1CC(=O)NCC1CCCC1NC(c1ccsn1)=O C=C(C)CC(C(=O)NC(c1cn(-c2cccc(OC(C)=O)c2)nn1)C)OC CCC(C)(C)C(=O)NC12CC1CN(C(C1CCCN(Cc3ccccc3)C1)=O)C2 c1(CN(c2nnc(-c3ccc(Br)s3)s2)CC)cccc(C)c1 c1(C(N2C(C)CC(CNC(c3c(CC)non3)=O)C2)=O)cc(C)c2[nH]cnc2c1 C1(NC(CN(C)C)=O)CCCC1NC(=O)C(CO)NC(=O)Cc1ccccc1 c1(C(C(=O)NCCSC)N(CC(C(=O)OC)O)C)cn2cnnc2cn1 c1(OC)cc(C(=O)NC2CC(CNC(=O)C(C)O)C(O)C2)c(F)cc1Br c1(C(N2CC(CNC(CCCn3c(C)nc(C)n3)=O)C2)=O)ccn2c1CCCC2 CCCC(CCNC(=O)CC1CC2(CC2)CN1C(C1CCCN1CC)=O)CCC C1(N(C(c2c(C)coc2)=O)C)CCCCC1NC(c1n[nH]cc1Cl)=O Nc1nccnc1C(N1CCCCC1CCC(=O)NCCN1CC2CCC1C2)=O Cc1nc2ccc(F)cc2c(C)c1C(=O)NCC1CCN1C(=O)C1=CCCC1C C(=O)(C(C)(F)C(C)(C)F)NCC(CC(C)C)NC(C1CCCC2C1C2(F)F)=O N1(C(CCC(C)OC)=O)CCC(NC(=O)CN(C)C(=O)C2CC2)C2(CCC2)C1 CS(=O)(=O)c1ccc(C(N2C3CCC2CN(C(C2CCCN2C=O)=O)C3)=O)o1 C1(CNC(CCOCC)=O)COCCN(C(C2CCCCNC2=O)=O)C1 C(=O)CC(CN(C(=O)OC(C)(C)C)CO)C(F)F.N(C(=S)NC(C)C)C(COC)C N1(C(c2n(CC)ncn2)=O)CCC(C2CC2NC(C2CN(C(N)=O)C2)=O)CC1 C1(NC(c2n(CC)ncn2)=O)CN(C(c2ccn(C3CC3)n2)=O)CC1SC C1(C(=O)NC2CCC(F)(F)C2)CC2CCC1N2C(c1cccc(Br)c1F)=O N1(C(CSCC(=O)OC)=O)CCC(NC(C2CC2CC(C)C)=O)C(C)(C)C1 N1(C(C=CC)=O)CC(CNC(c2sc(=NCC)[nH]c2C)=O)CCC1C N1(CC(n2cc(-c3ccc(CC)cc3)nn2)C)CCC2CCC(C1)S2 C#Cc1ccccc1C(N1CC(NC(c2cc3sccc3s2)=O)C(C#N)C1)=O c1(CC(=O)NC2CN(C(C(CN(C)C)O)=O)C2)cccc(Cl)c1F c1(C(=O)NCC=CCNC(c2c(CCC)occ2)=O)cc(C)nc(COC)n1 N1(C(c2cnc(C(=O)OC)s2)=O)CCCCC(NC(C2(C)CCCC2C)=O)C1 C(=O)(CCCCCCN=[N+]=[N-])N1CC2N(C(c3c(C)cc(F)cc3)=O)C(C2)C1 c1(OCCNC(=O)NCC2CCCOC2)cncc(Br)c1 C1(CN(C(CC2(NC(C)=O)CC2)=O)C)CCCN(C(c2cc(Cl)no2)=O)C1 c12ccc(cc1)C(=O)NC(C(C)C)CS2.C1(CC(=O)NCC=CC)CCCCC1 c1(SCc2cn(C)nc2O)ccc(C(=O)NC2CCN(C(C)=O)C2)cc1Cl C(=O)(CCCCC(=O)NC)N1CC(CNC(C(CCCC)O)=O)C1 c1(C(N(CC)CC2CCC(N(C)C)CC2)=O)ccc(N)c(-c2nn[nH]n2)c1 C1(CC(=O)NC2C(C)(C(F)F)C2)CC2(CC2)CN1C(c1ccc(C#N)o1)=O CCCCCC(CC)C(=O)NCCC1CCCN1C(c1ccc(CC)nc1C)=O Cc1nccnc1C(N1CCC(C)(NC(=O)CCCc2nc(C(C)C)no2)C1)=O C1(CNC(CCNC(=O)NC)=O)CC2CCC1N(C(C1(C3CC3)CCC1)=O)C2 c1(C(=O)NCC2CCC(NC(C(CC)(CC)OC)=O)C2)cnc2ccc(C)cn12 C1(C(=O)NCC(O)C(=O)NC2C=CCCC2)CC2CC1C(O)C2O C#CCC(C(=O)NCCCOCCN(C(=O)C(C1CCCCCC1)C)C)C1CC1 c1(NC=O)nc(CC(=O)NCC(CO)NC(c2[nH]cc(C(F)(F)F)c2)=O)cs1 C1(C(=O)NC2CC(NC(CSCCC(C)C)=O)CC2O)CCC([N+](=O)[O-])CC1 N1(C(c2c(C)nccn2)C(=O)NC(C)(C)C)C2CCC1CC(C)C2 C=CC(C)(CCOC)C(=O)N1CCCN(C(=O)COCC(F)F)C(C)C1 N1(C(C(C)NC(N)=O)=O)CCC2(NC(C3C4COCC34)=O)CCCCCC12 C(=O)(C(C)(C)CCNC(=O)OCC)Nc1cnc(OCC)[nH]1.C(C)(C)(C)O C(=O)(C1CCSc2ccccc21)NCC1(C)N(C(C(C=CC)O)=O)CC(F)(F)C1 C1(C(C)NC(=O)C(F)C2CC2)CN(C(=O)CC=C(Cl)Cl)CCO1 c1(C(C)(C)NCCCN2CCOC2=O)c(F)cccc1F Cc1ncc(CC(N2CC(CNC(c3ccccc3C)=O)C3CC23)=O)c(O)n1 c1(C(N2CC(NC(c3ccncc3)=O)CC23CCC3)=O)cc2c(Cl)cccn2n1 c1(NC(C2CC3CN(C(CCN(C(C)=O)C)=O)C2C3)=O)ccc([N+](=O)[O-])c(C)c1 CC1CN(C(=O)CCF)CCC1NC(=O)CS(=O)(=O)Cc1ccc(C#N)cc1 c1(CC)nc(OC)cc(N2CCC(C)(NC(c3cnns3)=O)C2)n1 C1(NC(C2(COCC)CC2)=O)CC2CCC(C1C)N2C(C1CC2CCCC12)=O c1(C(=O)NCCC(=O)NCCCCCC=C)c(C)ncnc1C C(=O)(C1(C)CCc2ccc(C)cc21)NCCNC(C12OCC(CC)(C1)C2)=O N1(C(=O)Nc2cc(C(F)(F)F)n(-c3ccccc3)n2)CC(CO)C(C2CC2)C1 C1(NC(COC)=O)CCOCC1NC(c1ccnc(C(N)=O)c1)=O N1(C(CCN(CCC)C)=O)CCOC(CCNC(c2cn(CCC)nc2C)=O)C1 N1(C(c2c(C)ccnn2)=O)CCN(C(c2ccn(C)n2)=O)C2CCCCC12 c1(C(=O)NCCCCn2cc(C(CC)O)nn2)ccc(OC)c(F)c1CC CCC(C(=O)N1CCC(C(=O)NOC(c2cccnc2)C)(OC)C1)C(C)(C)CC C=CC1(CC(N2CCCN(CCNC(c3cncnc3)=O)CC2)=O)CCCCC1 N1(C(c2cc(CC)on2)C(=O)NCC=C)CCCCCC1c1ccncc1 CN1C(=O)N2CCC(C(=O)NCCN(C(C3(c4cccnc4)CC3)=O)CC)C1C2 C1(CCCC)CN(C(=O)CC2CC(=O)NC2=O)CCN1C(c1cn(CC)cn1)=O C1(CNC(C=COCC)=O)CC(C)(C)CN1C(c1cnn(C)c1N)=O Cc1c(Br)cc(Cl)c(NC(C2(C3CC3)CNC2)=O)c1Cl.N12CCCC1C2 C1(NC(C2C(C)C2C)=O)CC2CN(C(C3CCCN3C=O)=O)CC12 C1(C(=O)NC2(C#C)CC2)COC2(C1)CN(C(c1n[nH]c(O)n1)=O)C2 c1(C(=O)NC2C(OC)CN(C(c3cc(C(F)F)no3)=O)C2)cc(C)ccc1F C1(CNC(C(C)OCCCC)=O)CC(F)(F)CN1c1nc(N(C)C)nc(=N)[nH]1 C1(C2CCN(C(=O)Cc3ccncc3Cl)C2)(NC(c2cc(C)c(C)nc2)=O)CC1 C1(CC(=O)N(CC(=C)C)C)CCN(C(c2cc(CC)oc2C)=O)C1(C)C c1(C(C)Nc2csc(N3CCOCC3)n2)cc(F)cc(Br)c1 c1(C(=O)NCC2N(C(C(C=C=C)C)=O)CCCC2)cc(O)nc2[nH]c(=N)ccc12 C(=O)(C(F)(F)C1=CCOCC1)NC12C(CN(C(CC(=O)NCC)=O)C1)CCC2 c1(C(N2CCCCC(NC(C3(C)ON=C(C)C3)=O)C2)=O)cc(C)c(F)cc1Cl c1(C(=O)NC2C(CNC(c3c(C)cc(CO)o3)=O)CCC2)cccc(F)c1N c1(OCC)ccc(C(C)NC(c2cnn(C3CC3(F)F)c2)=O)cc1 c1(CNC(C2(CCC)CC2)=O)n[nH]c2c1CN(C(=O)CC1CC(CC)=NO1)CC2 C(=O)(C1CCCn2nccc21)NC1CCN(C(c2n(C)ncc2)=O)CC1CO O=C(C#Cc1cccc(F)c1)c1ccc(-c2nn[nH]n2)nc1 C1(NC(c2cnc(C3CC3)[nH]2)=O)CCCCC1NC(c1ccsc1Br)=O N1(C(C2OCCN(C(c3csc(C)c3C)=O)C2)=O)CCC(O)C(F)C1 C1(NC(=O)Nc2ccc(-c3cn(C)nc3)cn2)CCC2CCCC2C1 c1(C(C)C(=O)NCCCCNC(=O)Cc2cnoc2)ccc2c(c1)OCO2 C1(NC(CCc2onc(C)n2)=O)CN(C(c2cn(C3CC3)cn2)=O)CCC1C C1(CNC(CC(=O)NC)=O)COCCN(C(=O)C#CC2CC2)C1 c1(C(N2CC3N(C(C(C)Oc4ccccc4)=O)C3C2)=O)cc2cc[nH]c2cc1Cl c1(N(C)C)cccc(NC(=NCC2CC2(Cl)Cl)NCCOCC2CCCO2)c1 c1(C(N(C)CC2CCN(C(c3ccoc3Br)=O)C2)=O)cc(N)cc(O)c1 C1(NC(=O)CSc2ccncc2)CC12CCN(C(c1ccc(Br)c(F)c1)=O)CC2 C(C)(CCC(=O)NCC(CC1CC1)C(=O)Nc1cccnc1C1CC1)OCC CC(C)(C)C1=NOC(C(N2CC(CNC(C3CC4C=CC3C4)=O)C2)=O)C1 N1(C(COCC(=O)OC)=O)CC2C3CCC(C2C1)N(C(=O)C(C)OCC(C)C)C3 C1(CCNC(C=C(C)C(F)F)=O)CC2CCC(C1)N2C(=O)CCOC1CCC1 Cc1ccc(-c2cc(C(N3CCN(C4CCN(CC=CCBr)CC4)CC3)=O)on2)cc1 c1(C(N2CCC(NC(C=CC=CC)=O)C2C(C)C)=O)ccc(=O)n(C)n1 c1(OCCn2c(COC)nnc2-c2ccc(O)cc2)ccccc1C C(=O)(CS(=O)(=O)CCOC)NC1CCN(C(C(C=C)(C)O)=O)CC1F Cc1oc(C(C)C)nc1C(N1CC(n2cc(C(n3cncn3)C)nn2)C(C)C1)=O c1(CCC(=O)NC(CC)CNC(=O)CCc2cn[nH]c2)ccc(C)cc1 C(=O)(C(CC1CCC1)NC(=O)C(C)=C1CC1)N(CC(COC)C)C c1(C(=O)NCC2(NC(c3cc(C(=O)OC)no3)=O)CCOC2)c(F)cccc1F c1(OCC)ccc(CC(=O)NC2CC2C(=O)NCCC(C)SC2CC2(F)F)cc1 CC(C)C(O)C(=O)N1CCC(OCCCNC(C2(C(=O)OC)CC2C)=O)CC1 C(CCCC(=O)N=c1ccn(CCNC(C(C)(C)C)=O)[nH]1)NS(N(C)C)(=O)=O C1(NC(C(C2CCOCC2)OC)=O)CCCC1CNC(C1(F)CCC1)=O C1(CNC(c2cc(OC)ncc2-c2cccnc2C)=O)CCCN2CCCCC12 c1(-c2cn(CCNC(=O)Cc3ccccc3)nn2)c(F)cccc1Br C1(CNC(CC(CNC(c2ccc(C)nc2C)=O)OC)=O)CCC2(CC2)CO1 C(=O)(C(C)(F)Cc1ccccc1)NCC(C)N(C(C1C(CC)C1)=O)C c1(N2CCC(CCOC)C2)cc(NCc2cc(C3CC3)no2)nc(C)n1 C(=O)(CS(=O)(=O)CCCC)NC1CN(C(C(F)=CCC)=O)C(C)CC1 C1(C(=O)NCCC(C)NC(C2CCN2C2CCCC2)=O)CCC=CCC1 N1(C(c2c(N)ccc(Cl)n2)=O)CCc2nc(CNC(=O)CCC3CCC3)sc2C1 C=CCC(C)(O)C(=O)N1CC2CC1(CNC(c1ncn(C3CC3)n1)=O)C2 c1(NCCC2CCN(NC(COCC(=C)C)=O)CC2)nc(C)nc(O)c1C C12(NC(c3cc(C(C)=O)oc3)=O)CCCCC1CN(C(=O)CC1(C(F)F)CC1)C2 C12CCC(C1)CC(=O)N1CC(C1)O2.c1scnc1Cl.CC(C)(C)OC=O.C1CN1 CC1CCCn2c(C(=O)NC(C)CCNC(=O)CNC(c3ccncc3)=O)cnc21 CCC(CC)C(C(=O)NCCN(C)C(c1ccccc1)C)CC(=O)NC1CCCC1 C1(CC=C)(NC(C2CC(Cl)(Cl)C2)=O)CCN(C(=O)Cc2ncncc2Cl)CC1 c1(C(N2CC(NC(C3CN(C)C(=O)N3)=O)C(C)(C)C2)=O)ccnc(S(N)(=O)=O)c1 C12(C(=O)NCCC(=O)NCC(COC)O)C=CC(CC1)C2 C1(C(=O)NCC(CCOC)NC(=O)C(C)C(=O)OC)CC2(CCCCC2)C1 C(C)(C(CC(=O)NC1CC(C(C)C)C1)NC(C1CCOC1(C)C)=O)OC C(=O)(CC(CC(C)C)NCC1CCC(c2nc[nH]n2)O1)OCC CC(C)C(F)(F)CC(=O)N1CCC(NC(c2ncc(F)cc2F)=O)C(F)C1 C(CC(=O)NCC1(CN=[N+]=[N-])CC1)(C(F)F)NC(c1nc(C)sc1C)=O c1(OCC)ccc(NCC(=O)NC23CC(NC(C4(C#N)CCCC4)=O)(C2)C3)cc1 CC1CCC(C(=O)NC2CCCC2NC(c2cc(Br)sn2)=O)C1 S(=O)(=O)(c1ccc(F)cc1)NC(CN1C(CS(C)(=O)=O)CC(F)(F)C1)=O C12(NCc3n(C)nnn3)CCC(C(N3CC4C(C3)C4(C)C)=O)(CC1)C2 C1(C(=O)OCC)CCN(C(c2ccc(C(F)(F)F)cc2OC(C)=O)=O)C2(CC2)C1 C(CCCCC(=O)N1CC(C(C)C)C1C(C)C)NC(c1cnc(CC)nc1)=O c1(OC)cc(N2CCCC(CNC(C3(N(C)C)CC3)=O)C2)ccc1[N+](=O)[O-] C12(NC(Cc3ccc(CC)cc3)=O)CCCC1N(C(C1(C)C=CCCC1)=O)CC2 c1(C(=O)NCC2(C)N(C(c3ncc(OC)cn3)=O)CCC2)ccc(C)c(Cl)c1F C1(NC(c2cn(CC=C)nn2)=O)CCCCC12CCCN(C(C1(C)CC1)=O)C2 C1(CC(=O)N(CCOC)CCNC(c2ccccc2)=O)CCC(O)CC1 C1(N(C(CCc2cn(C)nn2)=O)C)CCCC(NC(=O)CN2CCCNC2=O)C1 C12(CC)COC(C(N3CC(CNC(c4ccnc(N(C)C)c4)=O)CC3C)=O)(C1)C2 N1(C(C2CC(OCC)C2)=O)CC(C)CN(C(c2ccc(CC)c(C)c2)=O)C(C)C1 c1(C(=O)OC)cccc(CC(C(=O)NC(CO)C(C)NC(=O)C(OC)OC)OC)c1 Cc1nscc1CC(=O)N(CCCNC(=O)C=CBr)CC1CC1 C(=O)(CCCCN(C)C(C1C2CCCC12)=O)N(CC)Cc1ccc(CC)o1 C1(OCC(=O)NCC(CO)NC(c2n[nH]cc2Br)=O)CCC(F)(F)CC1 c1(CC)ccc(Br)c(C(=O)NC23CC(C2)N(NC(c2ccc(C)cc2F)=O)C3)c1 c1(C(=O)NC2C3CN(C(CC(C)OC)=O)CC32)ccc(F)c(Cl)c1 C1(C)(CNC(C2C(CCC)CCC2)=O)CSC(C)=N1.N12CSCC1C2=O C(=O)(C(CCOC(C1CC(N(C)C)C1)=O)N(C)C)N(C)CCN1CCCCC1 c1(C(=O)NCC2(NC(C3CC(CCC)C3)=O)CC2)ccc(CC)cc1O N1(C(CC2CC(OC)C2)=O)CCC(CN(C(=O)CCc2ccc(C)o2)C)C1 c1(N(C)CC2CCN(C(=O)C=Cc3ccccn3)CC2)nc(Cl)nc2[nH]ccc12 Cc1cc(NCC(=O)NC(=O)NC(CCCC(C)C)C(=O)O)cc(C#N)c1 C1(NC(c2c(CC)[nH]nc2Cl)=O)CCCN(C(c2ccn(C)c2C)=O)CC1F CC(C(=O)NC(C)(CNC(=O)C=CC1CCC1)C1CC1)NC(N)=O C1(NC(C(CC)OCC)=O)COCCN(C(c2cocn2)=O)C1 CCN=c1cc(C(=O)NCC2CC(NC(=O)C(n3nc(C)cc3C)C)C2)cc[nH]1 N1(C(C2C(OC)CC2)=O)CCC(C(=O)OC2CCC(CC(C)C)C2)C1 c1(C(=O)NC23CC(CNC(C4CCCOC4)=O)(C2)C3)occ2c1CCCC2 C(=O)(C(O)CC(C)C)NCCC1(NC(c2c(C)n(C)cn2)=O)CC1 c1(C(=O)NC(C2(O)CCN(c3nc(C)cc(C)n3)CC2)C)cc2n(n1)CCOC2 Cn1cc(C(=O)NCCCC(=O)NC2COC(C(F)F)C2)nn1 c1(C(=O)NCC2CN(C(c3ccsc3Cl)=O)CCO2)c[nH]c2nc(F)ccc12 N1(C(c2cncc(C)c2)=O)CCC(CCNC(=O)COCCCF)C(F)(F)C1 c1(CC2(C(=O)NC3CC(NC(CCC#C)=O)C3)CC2)cccc([N+](=O)[O-])c1 N1(C(CC(C)OC)=O)CCN(C(=O)CCc2ccc(Cl)cc2Cl)C(C)C1 c1(C(=O)NC2CC3CC(NC(C4CC(=C)C4)=O)C3C2)cc(Cl)cc([N+](=O)[O-])c1O Cc1cccc(C)c1CCNS(=O)(=O)c1c[nH]nc1C(C)C N1(C(c2cccc(Cl)c2)=O)CCC2(C1)CN(C(C1CC=CCC1)=O)CCO2 C(CN=c1[nH]c(NC(CSC)C)nc(=N)[nH]1)(c1ccccc1Cl)N(C)C C1(C(=O)NCC(C)N(C(c2nc(C(C)=O)sc2)=O)C)CCCC12CCC2 c1(C(=O)NC2C(NC(=O)OC(C)(C)C)CCOC2)ccc(C#N)cc1N n1(CC(=O)NC2C(OC)CN(C(CC=C)=O)C2)nc(C2CC2)n(C)c1=O C(=O)(C(C)C(C)NC(=O)C(CCC1CCC1)NC(=O)CC1CCCCN1C)OC N1(C(C(C)C)=O)CCC12CN(Cc1cnc(Cl)cn1)C2 O=C(CCCCCCC(=O)C1CC1)NC1CCCC1NC(C1CC12CCC2)=O N1(C(C2(C)CC(C)C2)=O)CCCC2(C1)CN(C(=O)C1=NOCC1)C2 N12C(CCC1C1CC1)C(=O)NCCSCC2=O.O=C(CSC(F)F)N c1(OC)cc(N2CC(OCCNC(C3CCC(C)(CC)O3)=O)C2)ccc1[N+](=O)[O-] c1(C(=O)NC23CC(NC(=O)Cc4cc(C5CC5)on4)(C2)C3)cc2scc(Cl)c2[nH]1 CCCCC(C)C(=O)N1CCCC1(C(=O)NCc1ccccc1Cl)CC CC1CN(C(=O)CCCOc2ccccn2)CCCN1C(=O)CCC(C)(C)F CC1(C)CC2(CC(NC(=O)NC3CCCCC34CC4)C2)C1 c1(C(=O)NCC2C(NC(Cc3cn(C(C)C)nc3)=O)C2)cc(Cl)c(N)cc1F c1(SCC)ccc(C(N2CCCCC2CNC(=O)CN(C)CCO)=O)cn1 C(C(C)C(F)(F)F)N(C(C(Cc1ccco1)NC(C1N(CC)CC1)=O)=O)C c1(OC)cccc(C(=O)NC2CN(Cc3ccc(F)c(CO)c3)CC2O)c1Br C1(NC(C2C(CC)CCN2C(C2C3CC(=O)CC23)=O)=O)CC2(C1)CC(C#N)C2 c1(C(N2CC(CNC(=O)CC(F)(F)F)OCCC2)=O)ccc2c(c1)CCCC2 C(=O)(CCCN(C)N=O)N(CCC)CCNC(c1cccn1C1CC1)=O c1(CC)ccc(OCCC(=O)N(C(C)CNC(=O)C=Cc2sccc2C)C)cc1 c1(CCC(=O)NC2C(NC(C3N(C)C(=O)CC3)=O)C2)ccc([N+](=O)[O-])cc1Cl c1(C(C(=O)OC)NCc2cnn(C)c2C(F)F)ccc(OC)c(Br)c1 c1(C(=O)NC(C)CCCCNC(=O)CCCSC(C)(C)C)c[nH]c2nc(Cl)ccc12 Cc1ccc(C)c(C(N2CC=CC2C(=O)NCc2ccnc(O)c2)=O)n1 N1(C(c2c(C)ncs2)=O)CCOC(CNC(c2ccnc(-c3ccco3)c2)=O)C1 c1(CC)nn(C)cc1C(=O)NC1CC12CC(NC(c1ccc(C(C)C)nc1)=O)C2 C12(C(=O)N(CCN(C)C3CC3)C3CC3)CCC(CN(C(N)=O)C1)C2 c1(CCNC(C2CCN(C(C)C(=O)N(C)C)CC2)=O)ncc(Cl)cc1Cl C1(NC(=O)NCC(N2CCN(C(=O)CC(=O)NC)CC2)=O)CCCCCC1CC c1(C(N(CCNC(c2ccc(CC)nc2C)=O)CC)=O)cccc2ncc(C)n12 C(=O)(C1=CSCCO1)NCC(CC(C)C)NC(=O)Cc1cn[nH]c1 Cc1cc(F)c(C(C)C)cc1Nc1cn(C(C)(C)C)nn1 N1(C(CC2(C)CC(F)(F)C2)=O)CC(NC(C2C3COCC23)=O)CC2(CC2)C1 N1(C(c2ccc(N(C)C)cc2)=O)CC(C)(C)C(NC(=O)C2=C(Cl)CC2)C(C)(C)C1 c1(C(=O)N(C(C2CN(C(=O)Cn3ccnn3)C2)=O)C2CC2)ccc(O)c(F)c1F c1(OC)ccc(C(N2CCCC(CCNC(=O)C(F)C(C)C)C2)=O)c(C)c1 CC(C(=O)NOCC(N1CCCCC1CCCO)=O)n1ccnc1 N1(C(CN(C(C(CCCC)F)=O)CCC)=O)CC2CCC(O)C(O)C12 N1(C(c2cc(OCC)n[nH]2)=O)CCCCCC(NC(c2cccc(N)c2C)=O)C1 C1(CN(C(=O)C(N)=O)C)CC(F)CN1C(c1ccc(C2CCCOC2)cc1)=O Cn1cc(C=CC(=O)NC(C)(CNC(c2cc(O)nn2C)=O)C2CC2)cn1 C1(C)(CNC(c2c(C)oc(Cl)n2)=O)CCCN(C(C23CC(C(=O)OC)(C2)C3)=O)C1 C1(NC(c2ncn(CC)n2)=O)CC(CC(=O)NCC2(CF)CCC2)C1(C)C Cc1cncc(C(=O)NC2CCCC2C(N2CCOCC2CCO)=O)n1 C1(OC)COCCC1CC(=O)Oc1nc(C(F)(F)F)c(C)s1 c1(C(CC)(C)C)n[nH]c(=NCCCOCCOC)o1 C=C(C)CCCC(=O)NC(C)(C)C=CC(=O)NC1CCC(C)CCC1 n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CC(COC)C2(C)C)cc1O c1(C(C)OCC)nc(CC(=O)N(C)CC2CCN(C(=O)CSS(C)(=O)=O)C2)cs1 c1(CC(=O)NCC23CC(SC)(C2)C3)ccc2scnc2c1 c1(OC)c(C)cc(C(=O)NC2(C)CCN(C(C3(C(=O)NC)CCC3)=O)C2)cc1C C1(C(=O)NC23CC(CNC(c4ccco4)=O)(C2)C3)(OC)CCOC1 C(C(F)(F)C(F)F)OCCC(N1C(CNC(c2ncn(C)n2)=O)CC1)=O C1(CC)CCN(C(=O)CCCOC(C)C)CC1n1cnnc1 c1(N(C(C(=O)NC2CCCCC2)C2CC2C)CC)ccccc1C(=O)NC C1(NC(CCNC(C)=O)=O)CCOCC1NC(c1n[nH]c(C)c1F)=O N1(C(CC=C(C)C)=O)CCOCC12CCN(C(=O)CCc1cnc[nH]1)C2 C1(C(=O)NCCS(CC)=O)CN(C(=O)CSC)CC12CCC2 c1(C2N(C(N=c3cnn(COC)[nH]3)=O)CCC2)c[nH]c2ccccc12 CCCCCCCCCCC(c1nnnn1C1CCC1)NCC(C)CSC C1(C(=O)NCC2C(C)(Br)C2)CC12CCN(Cc1cc(C(F)(F)F)ccc1O)C2 C1(CNC(C2C(C)C2)=O)CN(C(=O)Cc2ccc(F)nc2)CCC12CCC2 N1(c2n(CCOC)c(-c3ncnn3C(C)(C)C)nn2)CCC2(CCO2)C1 C(=O)(C(CCCCC1CC1)N(C)CC1(C)CCCCC1)NCC(=C)C C1(CCC)C(=O)N(C(=O)OCC(c2ccccc2)CN2CCOCC2)CC1OC c1(C(=O)NC2Cc3cscc3C2)ccc(-n2cc(CNS(N)(=O)=O)nn2)cc1F C(c1ccccn1)=CC(=O)NC(CCCNC(c1ccc(CNC(C)=O)o1)=O)C N1(C(c2cc(C(C)=O)on2)=O)CCC(C)C(CNC(c2c[nH]nc2Br)=O)C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC2C(C)O)=O)cnc2sccc2c1 c1(OC)cc2cc(NC(=O)NN3CCC3C)[nH]c2cc1Oc1ccccc1 O=C(C1Cc2ccc(F)cc21)NCCCOCCNC(c1ncoc1C1CC1)=O N1(CC)CC2CN(C(C34CCC3CN(C(=O)C(n3nccc3C)C)C4)=O)CC2C1 N1(C(C(C=C=C)C)=O)CCC2CCN(C(c3ccc(C#N)cc3F)=O)CC12 Nc1c(F)ccc(F)c1C(N1CC2CCN(C(C3CCS(=O)(=O)N3)=O)C2C1)=O c1(C(=O)NC2C(NC(c3cc(SC)ncc3)=O)COC2)c(C)ncn(C)c1=O Cc1nc2cccc(C(=O)NC3CCCCC3NC(=O)C(C)OCC3CC3)c2s1 c1(CCNC(C2C(CNC(c3scc(C)c3)=O)OCC2)=O)cccc(O)c1 C(=O)(CCCC(C)=O)NCC(CNC(c1cc(CC)nn1C)=O)(C)OC c1(CC)c(C(c2nnnn2CC(F)F)NC(C)Cc2cccs2)cnn1C N1(c2ccnc(COC)n2)CC2(CCC2)C1c1cccnc1 C(=O)(C(O)P(C)(C)=O)NCC(C)NC(c1cc(C)sc1)=O C(CC(C)CC)(C(=O)N(C)Cc1ccnn1C)NC(C(C)=CCC)=O C1(C(N2CCC(C)N(C(c3ccnn3C)=O)CC2)=O)CCC2(CCOCC2)C1 c1(C(N2CCCC(NC(C(CC=C)C)=O)CCC2)=O)ccc2c(c1)C(=O)CCO2 C1(NC(CC(C)c2ccccc2)=O)CN(C(c2ccncn2)=O)CC2CCCC12 Cn1nccc1C(CO)NC(=O)C(CC1CCCC1)NC(=O)C(F)C1CCCC1 Nc1ccc(F)cc1C(=O)NCC1CCC(NC(=O)CC2CCC2(F)F)C1 C1(CCNC(Cc2n(C)cnc2)=O)CCN(C(c2ccsc2)=O)CCC1(F)F N1(C(c2c(C)cccn2)=O)CC2CC1CN(C(=O)CC=CC(C)(C)C)C2 c1(C(N2CCC(CNC(C3(C4CC4)CCC3)=O)C2)=O)cc(F)ccc1Cl c1(C(=O)NC2CC(OCCCC)C2(C)C)c(Br)nc2n1CCC2 C(C(O)C(=O)NCCCCC1(NC(=O)CN2CCCCC2)CC1)=CCCC CCC(CC(=O)NCc1cc(OC)ns1)N(C)C(c1nncs1)=O c1(C(=O)NC(C2(CNC(c3nn[nH]c3Br)=O)CC2)C)ccc(O)cc1 C(CCCC(=O)NOC1CCC1)N(C(C1C(=C)C1)=O)CCF C(=O)(C1CCCc2nccn21)NC1(C)CN(C(c2ccn(CC(F)(F)F)n2)=O)C1 Cc1nc2cccc(C(N3C(C)C4CC3C4NC(C3CCCCS3)=O)=O)c2[nH]1 c1(OC)ccc(C(C)NCC(C)C(C)(F)F)c(Cl)c1 c1(OCCNC(=O)Nc2sccc2Cl)ccccc1O CN1CCC2OCCN(C(c3c[nH]nc3-c3cccs3)=O)C2C1 C(C1c2ccccc2CCN1C(=O)CC1CCNC1=O)NC(c1n(C)cnc1)=O c1(C(=O)NCC(CC=C)NC(=O)C(C)Cc2ccco2)cnc2[nH]cncc1-2 c1(NC(CCCCN(C(c2nc(CC)oc2C)=O)C)=O)cnc(Cl)nc1C c1(OC)cc(C)cnc1C(=O)NCC1(C(C)NC(C2CCC(=O)O2)=O)CC1 c1(-c2nnc(N(CCC)C)n2CCC#N)nc2c(s1)CCC2 C1(C(CNC(CCOC)=O)(C)O)CCCN(C(c2ccoc2CC(N)=O)=O)C1 c1(OCC)ccc2c(c1)CC(C(=O)NCC(O)COCC(F)(F)F)CO2 c1(C(=O)NCCC2(NC(c3ccoc3)=O)CCC2)n[nH]c(C2CC2)c1Br C=CCCCCCC(=O)NC1CN(C(C2CCCCN2CCC)=O)CC1C N1(C(C(C)(CO)OC)=O)CC2(CC(NC(=O)CC3CCCCCC3)C2)C1 C1(C(=O)OC)CC(=O)N(C)C1C(=O)NC(C)CNC(c1cn(C)nc1C)=O Cc1nc(CC(=O)NC2(CC(=O)NC3CCC(N(C)C)C3)CCC2)cs1 CC1(C)COc2cc(C(=O)NC3CC(F)(CNC(=O)CCC4CC4)C3)nn2C1 C12CC3CCC1CC3C(=O)N2.C(CCCN(C)C)N(C)C(=O)OC(C)(C)C c1(OC)ccc(C(=O)OCCC(C)(C)O)cc1S(=O)(=O)NC1=NCCC1 Cc1ncnc(C(=O)N(CCNC(=O)CCS(C)(=O)=O)Cc2ccccc2)c1C N1(C(c2cnn(CC)c2C)=O)CCCC(NC(c2ccnn2C(C)C)=O)C1C C(CCNC(=O)NC1(CO)CC(O)C1)(C(C)C)NC(=O)OCC C1(CC(C)NC(=O)CCCNS(C)(=O)=O)CCN(C(C2COC(C)C2)=O)CC1 C1(C)(C(N(CC)Cc2cccnc2)=O)CCCN(C(C2CCN(C)CC2)=O)C1 c1(C(N2CCN(C(c3cc(CC)n(C)n3)=O)C(CO)C2)=O)c(C)cc(O)cc1O C1(C(=O)NC2C(C=C)COC2)CC(C)(C)CCN1C(=O)C=CC1CCC1 C1(CC(C)NC(c2ccc(NC)cc2)=O)CCN(C(=O)CC2CSCCS2)CC1 C#Cc1cc(C(N2CCC3(CC2)CC3NC(=O)C=C(CC)CC)=O)ccc1Cl C(=O)(C1CCCc2nncn21)NC1CCN(C(C2N(C)CCC2)=O)CC1CO c1(NC(C2C(Nc3ncc(C)cn3)C2)=O)cc(Br)ccc1I CC1CC(NC(=O)C=C(C2CC2)C2CC2)CN(C(=O)C(c2cccnc2)O)C1 N1(C(c2cc(CC)no2)=O)CC2CCCC2(CNC(C2(COC)CC2(F)F)=O)C1 Cc1cc([N+](=O)[O-])cc(C(N2CCC(O)(c3nc(C4CC4)no3)C2)=O)n1 N(C1CCCc2ccccc21)C(C1N(C(C2CNC(=O)O2)=O)CCOC1)=O O=[N+]([O-])c1cc(F)c2c(c1)CN(Cc1snc3ccccc13)CC2 c1(N(C)C)cccnc1C(=O)NC1C=CC(C(N2CCCCC2C(N)=O)=O)C1 c1(OCC)ccc(F)cc1NCc1ccc(F)c(OC)c1 C(=O)(C(O)CN1CCOCC1)NCC1N(C(C2CC(=C3CCC3)C2)=O)CC1 N1(C(C(C2(OC)CCOCC2)(F)F)=O)CC2(CCN2C(C23CCC(C2)C3)=O)C1 c1(OCC)ncc(C(=O)NCCOCCN(C)C(C23CCC(C2)C3)=O)cc1Cl N1(C(C(CC=C)C)=O)CCCN(C(=O)C2=CC(C)(C)C2)C(C)C1 n1(CC(=O)NCC(CC)(C)NC(=O)CN(C)C(N)=O)ccc([N+](=O)[O-])n1 C(c1c(Cl)cccc1Cl)=C(C(=O)NCCC(=C)CNC(=O)C(C)CC(F)F)C C1(NC(c2n(CC)nnc2)=O)C2CC1CN(C(=O)CC1COCCN1C(C)=O)C2 c1(C(N2C(C(C)NC(c3nocc3Cl)=O)CCC2)=O)cc(C(F)F)ncn1 C1(C(=O)NCCSC)CCCN1C(=O)C(C)NC(C)=O CCCCC(O)CCC(=O)NCC1CCC(NC(=O)C=Cc2ccncc2C)C1 CCC(CC)(C(=O)NC(C1CCCC1)CNC(=O)Cc1nc[nH]n1)OC Cc1cc[nH]c(=N)c1C(N1CCCC(N(C)C(C2CC2C(F)(F)F)=O)C1)=O N1(C(C2(C#N)C(C)(C)C2)=O)CCC2CN(C(c3csc(Cl)c3)=O)C2C1 C1(C)(CC(=O)NC2(c3ccc(F)cn3)CC2)CCN(C(C2C(C)(C)C2CO)=O)C1 C1(F)(C(=O)NCC2(COCC)CN(C(C(CC)N(C)C)=O)C2)CCCN(C)C1 CCC(C)C(C)C(=O)NC1CCCCN(C(C2C3CCC(=O)C23)=O)C1 C1(C(=O)NCC(N(C)C(c2coc(Cl)n2)=O)C2CC2)CC2(CCOC2)C1 C(=O)(C1=CCCCO1)NC1C(NC(C2C(C)CC2)=O)CCC1 C1(N(C(CCOCCC)=O)CC(C)C)CCN(C(C2CC2(F)Cl)=O)CC1 CCCCC(C(=O)NCC12CC(CN1C(C1COC(=O)N1C)=O)C2)C(C)C C1(OC)CC2(C1)CN(C(=O)C(CC1CC1)NC(=O)CC(C)(C)C)C2 C1(NC(C2(N(C)C)CCCCC2)=O)COCCN(C(c2cc(O)ncc2F)=O)C1 N1(C(C(C)C2CC2)C(=O)NC2CCCCC2)CC2COCC2(C)C1 c1(C(N2CCCC(F)(CNC(=O)Cc3ccsn3)C2)=O)oc2ccccc2c1Cl c1(C(=O)NC)nn(C)c(OC)c1C(=O)NC1CCC(=O)N1c1ccc(C)cc1 N1(C(C2C(C(C)(F)F)C2)=O)CC2(C1)CN(C(=O)CC1CC3(CC3)CO1)C2 c1(C(=O)NCCc2cc(C)cc(C)c2)ccc(Br)c(Cl)c1N c1(CC(=O)OCCCc2cn(CC(CC)O)nn2)noc(C)c1C#N Cc1nc2ccccc2cc1NC(=O)NC12CC(F)C1C2 C12(NC(C3N(C)CC(O)C3)=O)CCC(C1)N(C(=O)Cc1c(O)ncnc1O)C2 c1(C(C(=O)NC2(CC)CC2)N(C2(CO)CCCC2)C)ccc2c(c1)CCC2 C1(C(=O)NC2(CN(C(C(n3ncc(C)c3)C)=O)C)CC2)CC1C1CCC1 C(=O)(C1CCc2cccc(O)c21)NCC(CCNC(CCNC(=O)NC)=O)C C1(C(N(CCN(C(=O)Cc2cnnn2C)C)C)=O)CC2CC1C1CC21 CC(C)CC(O)C(=O)N1CC(O)CC1CNC(=O)C1=CCCC1C C1(NCCN2CCC(NC(=O)C3=CCCCC3)CC2)CCC2CCCCN12 N1(Cc2cccc(OCC)c2)CCCCC(NC(C2CC2(C)C)=O)C1 C1(C(=O)NCC(C)CCO)CCCN(C(=O)CCN(C)CCO)CC1 C=C(C)C(C)(O)C(=O)NCCC1(O)CCN(C(=O)CCNc2ccccn2)CC1 c1(C(C(=O)N(C(C)CN(C)C)C)C)c(I)cnn1-c1cccs1 c1(CNC(C(=O)NC2CC(C)N(C(=O)NCC(F)F)C2)=O)ccc([N+](=O)[O-])nc1 C1(C(=O)NC)CC(O)CN1C(=O)N(CCCCO)C(C)C C=CC(C)(CC)C(=O)NC1(CNC(c2cc(-n3cccn3)ccn2)=O)CCCC1 N1(C(C2CCSC2)=O)CC2CCC1C1CN(C(C3CCCCO3)=O)CC21 CCCC(CCC)C(=O)N1CCC(CNC(=O)C(F)CC2CCCCC2)C1(C)C N1(C(C(C)N=[N+]=[N-])=O)CCN(C)CC1CNC(C1CC2(CC2)CO1)=O c1(CC(=O)NCCc2cc(O)cc(Br)c2)ccc2c(c1)OCO2 C1(N(C)C(c2nocc2Cl)=O)CCCCN(C(c2ccn(CC(F)(F)F)n2)=O)C1 c1(OC)ncc(F)cc1C(N1CCC(CCNC(c2ccoc2C)=O)C1)=O N1(CCN(C(=O)C(C2CCN(C(c3cc(CO)[nH]n3)=O)C2)F)C)CCCNC1=O c1(NC(=O)NCCCNC(C(C)OC)=O)cc(S(N)(=O)=O)c(C)cc1C N1(C(=O)CCN2CCC2)CCC2CCN(C(=O)CC3CC(F)C3)C2C1 CCCC(CC)C(=O)N(CC(CC)NC(c1cc(NC(C)=O)ccc1C)=O)CC C(=O)(C(C)(F)C(=O)NCCN(C(=O)CN1CCCC1CO)C(C)C)OC c1(C(=O)NC2CCCC(NC(CCC3CCN(C)C3)=O)C2)ccc([N+](=O)[O-])[nH]1 C1(O)(CNC(CC(=O)N(C)C)=O)CCCN(C(C2CC(=O)OC2(C)C)=O)C1 N1(CC)N=C(C(=O)N2CC(NC(=O)CCOc3ccc(F)c(Cl)c3)C2)CCC1=O CN1CC(O)CC1(C)C(N1CC2(C1)CN(C(=O)CN1CC3CC3C1)C2)=O C(c1ccc(Cl)cc1F)=CC(N1CC(CNC(c2ccc(Cl)c(O)c2)=O)C1)=O C(=O)(C(C(C)OC)NC(c1[nH]ccc1C)=O)N1C(C)(C(=O)OC)CC1 C=C(F)C1(CC(=O)NCC2CCCN2C(C2(S(N)(=O)=O)CC2)=O)CCC1 c1(Nc2c(SC)occ2)ccnc(NC(C2CC(C)CN2c2ccncn2)=O)c1 N1(C(CC(C)(C)OC)=O)CCN(C(=O)CC2CC3(CCC3)C2)C(CO)C1 CC1=C(C(=O)N2CCC(O)(CNC(c3cc4ccsc4s3)=O)C2)CCC1 Cc1cc(C(=O)NCCCCCN(C)Cc2cn(Cc3cccnn3)nn2)co1 Cc1cncc(C(=O)NCCC2CCN(C(c3ccnc(O)c3)=O)C2)c1 N1(C(CCOCCOC)=O)CC2(COC(CNC(=O)CC3CC4(CC4)CO3)C2)C1 N1(C(C2CC(OC)C2)=O)CCOC(C)(CNC(C2(Cl)CC2(C)C)=O)C1 CCCCCCC(=O)NC1C=CC(CNC(=O)C(C)(CO)OC)C1 c1(OC)ccc(C(C)C(=O)NC(CNC(=O)C=CBr)C2CCCC2)cc1OC N(C)(C(=NCc1cnnn1C)NC(CC)CC)CC(C)Oc1cccc(OC)c1 c1(C(=O)NCCCCN(C(COCC(=O)NC)=O)CCC#N)cn(C)nc1O C(N=c1cc[nH]cc1[N+](=O)[O-])C1COCCN(C(=O)C(C2CCOCC2)F)C1 C1(NC(CC(=O)NCC)=O)C2CCC(C2)C1C(=O)N(CC(C)(O)C1CC1)C CC1CCN(C(C2CNC(=O)C2)=O)C1C(=O)NCCCN=[N+]=[N-] C12(NC(C(CC)C)=O)CCC(NC(c3cscc3C(F)F)=O)(CC1)C2 N1(C(COCC(=C)C)=O)C2CCC1CN(C(C1(OC(C)=O)CC1)=O)C2 CC(C)(O)CCCNC1(c2nnnn2C)CCC(CN2CCOCC2)C1 N1(C(CNC(=O)Cn2cncn2)=O)CCCN(C(c2coc(Br)c2)=O)CC1 N1(C(c2c(C)nsc2)=O)CCN(C(c2cncc(F)c2C)=O)CC1CC(F)F CC1CN(C(C2CCCC(O)C2)=O)CC1CC(=O)N(C1CC1)CC1CCCO1 C1(OC)(CNC(=O)CC(=O)N(C)C)CCN(C(c2ccccc2SC(C)C)=O)C1 c1(C(N2CC(C)C(CNC(=O)C(c3cscn3)N(C)C)C2)=O)cn2ccccc2n1 Cc1cccc(C(=O)NC2CC2NC(c2cc(C3CC(F)(F)C3)[nH]n2)=O)c1O N1(C(C2N(C(CCCOCCSC)=O)CC2)=O)CCC(O)(C(F)F)C1 C12(CC)CCC(C(N3CCCC(CNC(c4cnccc4C)=O)C3)=O)(CC1)CO2 c1(C(N2CCN(C(C(CC)(C)C)=O)CC2C2CC2)=O)cc(S(N)(=O)=O)c(Cl)o1 c1(C(N(c2c(C)c(Cl)ncn2)CC2CN3CCN2C(C)C3)=O)ccnc2ccsc12 C1(C(C2CCCC2)NC(CC)CNC(c2nocc2C2CC2)=O)CCC(C)CC1 N1(C(COCC(=O)OC)=O)CC2CCCC(N(C(=O)C(F)C3CC3)C)C2C1 N1(C(c2cc(C)sc2Br)=O)CCC2(C1)CN(C(=O)CC1COCCN1C)C2 c1(SC(C)CNC(=O)NC2CC2(F)F)nc2ccccc2s1 N1(C(CC(=C)Br)=O)CCN(C(c2ccc(N)c(O)c2)=O)CCC1C CCC(F)(F)C(C)(C)C(=O)N(CCCNC(c1cc2n(n1)CCO2)=O)C c1(C(=O)NCC=CCNC(C=CCCC)=O)cccc(OC)c1 c12cccnc1OCC(=O)NC(CN)CN2.C(=O)(C1CC1)C(=O)C(C)C.CSN N1(C(C2CCC(C)CC2)=O)CC2(C1)CN(C(=O)C(F)C(F)(F)F)CC2CO C(=O)(CC(C(F)F)C(C)(C)C)NC(C(C)C)CNC(c1nsnc1O)=O C1(CN(C(=O)Cc2ccco2)CC)CCCN(C(C2CCC(=O)C2)=O)C1 C(=O)(CC(C)(C)C(C)(F)F)NCC1C(C)CCN1C(c1ccc(Cl)cc1)=O C(=O)(C(C)C(O)C(C)CC)NCCOCCC(N1CCCC(=C)C1)=O C1(CC)C(NC(c2cnc(C(F)(F)F)cn2)=O)CCN1C(=O)C=Cc1cnc[nH]1 c1(SC)nc(O)c(C(=O)OC(c2ccc(F)cc2Cl)C)cc1C#N CC1=C(C)CC(C(=O)N(C2C3CN(C(c4ccc(O)nc4C)=O)CC23)C)CC1 c1(C(=O)NC(C(=O)NCC2C(OCC)CC2)C2CC2)cnc(Cl)s1 Cc1cc(C)n2ncc(C(N3CCC4(CC(NC(=O)C5=CCC5)CO4)C3)=O)c2n1 c1(C(N(C2CN(C(=O)C=CC(F)(F)F)CC2F)C)=O)onc2c1CCCC2 C(=O)(C1=NOC2(CCOC2)C1)Nc1cccc(NC(C(F)OC)=O)c1 c1(NC(C)Cc2ccco2)ccc(S(=O)(=O)NCCC2CCCN(C)C2)cc1Br Cc1ccc(C(N2CCCC(C3OCCC3C(=O)O)C2)=O)cc1[N+](=O)[O-] c1(C(=O)NCC2CCCN(C(C3(C)C=CCC3)=O)C2)ccnc(Cl)c1O Cc1cc(COCC(=O)NCC2(F)CN(C(C3CC4CC3C4)=O)C2)no1 c1(-n2cc(-c3c(C)con3)nn2)cccc(CCNC(C2CCS(=O)(=O)N2)=O)c1 S(=O)(=O)(CC(=O)N1CCCC1C1(C(=O)NCC(CC2CC2)CO)CC1)N(C)C C(C(C)(C)C(C)(F)F)(c1nnnn1C(C)(C)C)NCCc1ccnc(C)n1 c1(COC)nn(C)cc1C(=O)NCC1(F)CN(C(=O)CCn2ccccc2=O)C1 C1(C(C)(C)C)CN(C(c2csc(-c3ccoc3)n2)=O)CCC1CC(=O)O N1(C(C(CC)N(C(=O)CCc2ccsc2)C)=O)CC(C)C(O)C(C)C1 c1(C(c2nnnn2CCS)NCC(=C)C)cccc2ccncc12.C1(C)CCCO1 C1(CNC(c2ccc(CCC)s2)=O)CC2CCC1N2C(c1cc[nH]c1)=O O=C(C1=COCCC1)NCC1CCC(C(=O)Nc2ccc(Br)c(F)c2)C1 c12ccccc1C(=O)NC(=O)COCCO2.C1(NCCO)CN(CCC(=O)O)C1 C1(N(C(CSSC)=O)CC)CCCN(C(C2CCCN(CC(F)F)C2)=O)CC1 C1(=O)CC(C(C)CC)N1C(C=C)(C)C.C(=O)(C(C)(O)CCN(C)C)NC1CC1 C(=O)(CCCCCNC(=O)C1CC1)NC(c1nnc(O)o1)C N1(C(c2c(CC)ccs2)=O)CC(NC(=O)C2=CCCSC2)CC1(C)C C1(C)(C(=O)NC(COCC)(C)C)CCCN(C(c2cccc(F)c2)=O)C1 C1(NC(CN(C)C)=O)COC2(CCCN(C(=O)COc3ccc(Cl)cc3Cl)C2)C1 O=C(CC1OCCc2sccc21)N1CCc2sc(Br)cc2C1 C1(NC(c2n(CC)ccn2)=O)CN(C(=O)CCn2nc(C)nc2C)CC2(CC2)C1 N1(C(CCNC(=O)CO)=O)CC2CC1CN(C(=O)CC1CCCC13CC3)C2 c1(C(N2CCC(C(N3CC(OC)C(C)(C)C3)=O)(CC)C2)=O)ccn2nccc2c1 c1(OC)ncccc1C(N1CCCC1C(C)NC(=O)CCOc1ccccn1)=O c1(CNC(CCC#C)c2ccccc2)cc(C)ccc1Br N1(c2cc(C)nc(NC3CC4(C3)CC(C)C4)n2)CC2CCCC(C1)N2C C1(NC(COCCCOC)=O)CN(C(c2c(C)cnn2C(C)C)=O)CCC1O C(=O)(C(C)(C)C1CCOC1)N(CC(=O)N(C1CC(CC)C1)C)CC O=[N+]([O-])c1nn(-c2ccc(F)cc2)nc1OCc1ccc(C(F)F)cc1 C1(C#CC(=O)N(C(C)CC(=O)NC(C)C(C)n2cccn2)C)(CC)COC1 n1(C(C(=O)N(CC(CC)NC(=O)C(=Cc2cccs2)C)CC)C)ccnc1C C(CCCCC(=O)N1CCOC(C)(CNC(=O)CCc2cccc(C)c2)C1)OC C1(C(=O)NCC2CC=CCC2)CCCN(C(C2CCC(O)C2)=O)C1 C1(CC(N2CC(CC)(CC)C2)=O)CCCN(C(=O)CSS(C)(=O)=O)C1 c1(CN2CCN(C(C3CC3c3ccc(Cl)cc3)=O)C3C2C3)ccc(Br)c(F)c1F c1(C(=O)NCCC2(NC(C3N(CC(C)C)CCC3)=O)CC2)cnc(O)c(Br)c1 c1(CC(=O)N(CC(=O)NC(COCC)C)C(C)C)occc1C C(CN=c1[nH]c(=NCC(C)c2c(C)noc2C)c2ccc(OC)cc2[nH]1)OC N1(C(C(C)N(C)C)=O)CCOC2(CCC(NC(=O)C(C)n3cccc3)CC2)C1 C(CN=c1nc2sccc2c(NCC2CCCC2(F)F)[nH]1)(C1CCCC1)OCC Cc1nc(C(N2CC3CC(NC(=O)C(C)(C)F)C2C3)=O)c(=O)[nH]c1C CC1(C)COC(C(=O)NC(c2ccc(F)cc2)(C)CNC(=O)C(F)=CCCF)C1 Cc1ccccc1NC(=O)C(N1CCC(Oc2ccc(Cl)cc2)C1)C c1(CC)csc(C(c2nnnn2C(C)C(=O)OC)NCCOC(C)C)n1 c1(C(N2CC(CCC=C)(C(=O)NC(C)CCC)C2)=O)ncc(F)cc1C C1(O)(CC(=O)NCC2C(NC(C3(CC#N)COC3)=O)CCCC2)CCCCCC1 N1(C(C(C)OC)=O)C2CCC1CN(C(c1cnns1)=O)C2 C1(C(=O)NCC2C(NC(c3cncc4c[nH]nc34)=O)C2)CC12CCC(F)(F)CC2 C(=O)(C(C)(F)C(F)(F)F)NCC1CC(OC)CN1C(=O)C=Cc1ccncc1 Cc1ccc(C)c(NC(C2CCC2CNC(c2c(C)nsc2C)=O)=O)c1 c1(C(N2C(C)CCC(NC(=O)CC3CCN(C)CC3)C2)=O)ccc(C#N)cc1O N1(C(CCCC)=O)CC2CCC1C1CN(c3ncnc4cc(C)[nH]c34)CC21 C(CC(C(=O)N1CCCC1C(=O)N(C)C)NC(c1cc(Cl)n[nH]1)=O)SC c1(NC(C2CN(C(C3CCN(C)C3)=O)CC(F)C2)=O)cc(F)c(Cl)nc1Cl C1(CNC(C(C)OCCC=C)=O)CC(CC(N2CC=C(C)CC2)=O)C1(C)C c1(OC)ccc(NCCNC(c2cn(C)nc2SC)C)cc1.C1CO1 c1(C(=O)NC(COCCC)CO)cccc(NC(c2cc(SC3CC3)n[nH]2)=O)c1 c1(C(N(C)CC2(CNC(=O)C(F)C3CCOC3)CC2)=O)c[nH]c(=N)o1 C1(n2cc(CCSCC)nn2)CCCN(C(=O)C(C)Cc2ccnn2C)CC1 N1(C(CC2C(C)CCN(C(=O)CN(C3CCC3)C)C2)=O)CCC2(CC1)CC2CO C1(CNC(=O)C(F)CC2CC2)(CO)CCCN(C(=O)CCC23CCC(CC2)C3)C1 CCC(CCC(=O)N1CC(O)C(O)C1CNC(c1conc1C)=O)OC C(CN=[N+]=[N-])(C(=O)N1CCCC(C)(O)C1)NC(c1c(COC)cco1)=O CCC(CC(C)C)C(=O)NC1CN(C(=O)CCc2cccn2C)C1 C1(C(=O)OCC)CCN(c2nnc(CC)n2CCCS(C)(=O)=O)CC1.CCCCSC Cc1c(C(=O)NCC2CCCCN2C(=O)Cc2cnnc(O)c2)cnn1C(C)C c1(OC(C(=O)NCC(CC)NC(C2(CO)COC2)=O)CC)cccc(Cl)c1Cl C1(NC(C(C)Sc2n[nH]c(O)n2)=O)C(=O)OC2CCCC12 Cc1ncnc(C(N2CC(O)CC2CC(=O)N(C(C)CO)C)=O)c1C C(=O)(CC(O)C(C)(C)C)N1C(C(CNC(CCC)=O)(C)C)CCCC1 c1(CNC(C=CC2(C)COC2)=O)nnc2n1CCN(C(c1ccc(Cl)o1)=O)C2 C#CC(C)(C)C(=O)NCCC1CCCCN1C(=O)CCCF C(=O)(C#CC1CCCCO1)N1CCN(C(c2ccc(CC)[nH]2)=O)CC1C(C)C Cc1cccc(C(=O)NCc2ncccc2CNC(C2CNC(=O)N2C)=O)n1 CCCCCC(C)CC(=O)N1CCN(C(C2CC(C)(F)C2)=O)C(C2CCCC2)C1 N12CCCC(CO)(C1)NC(=O)COCC2=O.C1(N(C)CO)CCN(S(C)(=O)=O)CC1 C1(CNC(OCCOC)=O)COC(C(F)(F)F)CN1C(=O)CC1(O)CCOCC1 c1(CCC(=O)NCCC(CNC(C(C)CC2CC2)=O)O)ccccc1F C1(NC(CSCCOC)=O)CCC2(CCN(C(C3Cc4cccnc4C3)=O)C2)C1 c1(CNCCOc2ccc(CC(=O)O)cc2)nnc2n1CCOC2 Cc1cc(N2CC(C)C(C)C2)ncc1S(=O)(=O)N1CCC(CCCO)CC1.N(C)C c1(C2CC(C(=O)NC3C(NC(=O)CCC4CCCCO4)C3)C2)cccc(Cl)c1 C(=O)(C(C(C)(C)C)N1CCNC1=O)N1CCC(OC)(CNC(C2CCS(=O)(=O)C2)=O)C1 N1(C(c2n[nH]c(C)c2C)=O)CCN(C(c2cnn(C3COC3)c2)=O)C(C)C1C N#Cc1nc(=NC2C3CC2CN(C(c2cc4ccoc4s2)=O)C3)cc[nH]1 C(=O)(CC(C)(O)C(F)(F)F)NCC(CNC(c1n(CC)ncn1)=O)(C)O c1(C(N2CC(CNC(C3C(C)C3)=O)N(C)CC2)=O)nccn2ccnc12 Cc1onc(C(F)(F)F)c1C(N1CC(O)(CNC(=O)C#CC2CC2)C1)=O Cc1ccc(C(=O)NC(C2CCCN2C(C2CC(=C(F)F)C2)=O)C)cc1O c1(C(N2C(CNC(CSCCC(C)C)=O)CCCC2)=O)c[nH]c2ccncc12 Cc1cc(C(=O)NCc2cc(C(=O)N(C)CC3CCCCO3)n(C)n2)ncc1N C(C)(CCCCNC(c1ccc(OCCC)cc1)=O)NC(C(CC)=CC)=O CCC(C)(C(=O)NCC1CC(F)CN1C(c1cc(CN(C)C)c[nH]1)=O)C(F)F C#CCCCC(=O)N1CCOCC1CNC(=O)CC1(NC(=O)OC(C)(C)C)CC1 Cc1nn(C)cc1S(=O)(=O)N1CC2C(NC(c3ccc(F)nc3C)=O)C2C1 c1(C(=O)NC2(C)CC(NC(C3CN(CC(C)C)C(=O)C3)=O)C2)ccn2ccsc12 N1(C(c2c(C)nsc2)=O)CC2CCC1CC2NC(C1CC2CC2C1)=O Cc1c(C(F)F)n[nH]c1C(=O)NCCCOC(F)F CC1CC(C(=O)NCC(O)CCC2CC2)N1C(=O)COC1(C)CCC1 C1(CNC(=O)C=C(Cl)Cl)CN(C(=O)COc2cccc(F)c2)CCC1(F)F C(=O)(C(O)CC(F)(F)F)N1CC(C(C(=O)Nc2ccc(OC)nc2)O)C1 N1(C(CC2CC(=O)NC2=O)=O)CC2CC1CN2C(c1ccccc1)=O c1(CCOC)nc(=NCC(C)N(C(C(=O)NC(C)C)=O)C)s[nH]1 CCCC(C)CC(=O)NCCCC(C)NC(=O)Cc1c(C)nn(CC)c1C C1(CCNC(=O)C2=CCCOC2)CN(C(C23CCCC2CCC3)=O)CCS1(=O)=O c1(C(=O)NCC23C(CN(C(CCCCC#C)=O)C2)C3)scc2c1CCCC2 C1(CC(=O)NC(c2ccccc2Cl)COC)CCC2(CCC2)CO1 C=C(C)CCCC(=O)NC1(C)CCN(C(=O)C(C)(O)C=C)C1 c1(C(N(C2CCN(C(C(C3CCOCC3)OC)=O)C2)C)=O)cc(Cl)ccc1F C(=O)(CS(=O)(=O)CCOC)NC1CN(C(CC2(C(=O)OC)CC2)=O)C(CC)(CC)C1 N1(C(C(CC)C)=O)CC(NC(c2cnc(C(F)F)nc2)=O)CC1C c1(CC)cncc(C(c2nnnn2-c2ccc(OC)cc2)NCC(C)(C)C)c1 C(=O)(CCC(=O)c1cccnc1)NC(C)(CNC(=O)C=Cc1ncc[nH]1)CO c1(CC(C)C)ccccc1C(C)OC(=O)CSc1nnnn1C Cc1cnc(NC2CN(C3CCOCC3)C2)c(S(=O)(=O)N2C(C)CCC2C)c1 Cc1cnc(C(=O)Nc2cccc(NC(c3ccn(C)c3)=O)c2)nc1 N1(C(C(C)=CC)=O)CC(NC(=O)CC2CCCC(C)C2)C2(CCOCC2)C1 c1(C(=O)NCCCN2C(c3cccc(C)c3)C(=O)NCC2)cnn2c1OCC(O)C2 C1(C)(CNC(CCN2CCN(C)CC2)=O)CCCN(C(c2cc(C#N)no2)=O)C1 c1(N(C)C)cccc(OCC(=O)Nc2cccc(NS(N)(=O)=O)c2)c1 c1(C(=O)NCC(CNC(=O)C=C(C)C)OC)cc(N)ccc1C c1(CCC(=O)NC2C(NC(c3c(C)cno3)=O)CCOC2)cnc2n1CCOC2 C12(C(N(CCCCC=C)C)=O)CC(CO1)N(C(C1CCOCC1)=O)C2 C1(C(=O)NCCSC(C)C)(NC(=O)CC2CCSC2)CCN(C)C1 N1(CCC2CC2)CCCSCC1.CC1CCN(C(=O)CCn2cc(CC)nn2)C1 CCC(C)C(C)C(=O)NCCCCNC(=O)COc1cccc(F)n1 c1(C(N(CC(=O)N(C)CC)CC#C)=O)ccc(F)nc1 C12(C(N3CC(OC(C=C)=O)C3)=O)CC(CN1C(C1CCCC(=C)C1)=O)C2 C(=O)(C(CC(C)C)N(C)C)N1CCC(CN(C(C2CNC(=O)C2)=O)CC)CC1 c1(C(N2CCCC(N(C(c3ccc(C)n3C)=O)C)C2)=O)cnc(P(C)(C)=O)cn1 C1(CNC(=O)CCCC2CC2)CCCN(C(=O)C=CCNC=O)CC1 C=CC(CC(=O)NC(C)CN(C)C(C1(CC)CCOCC1)=O)c1ccccc1 c1(C(=O)NC(C(C)C)C2CCC2)n[nH]c2c1CN(C(c1c[nH]nc1C(C)C)=O)C2 N1(C(C(C)=C2CCC2)=O)CC(NC(=O)C(F)(F)CO)C(C)C1 C1(C(C(=O)OCC)Cc2ccc(C)cc2)CCN(C(c2cnc(S)nc2)=O)CC1 CC(CCC(C)(C)C)C(=O)N(C)CCOCCCNC(=O)Cc1cnsc1 C(C1=NOC2CCCCC12)n1cc(-c2cc(C(=O)OC)c(F)nc2)nn1 c1(C(N(CCC(C)NC(c2ccc(C3CCCO3)[nH]2)=O)C)=O)csc(=N)[nH]1 c1(C(N2C(CNC(CN(CC)CC)=O)COCC2)=O)csc2nccn12 CCC(C)(C)C(=O)N(C(CNC(=O)CC1CCCC12CC2)C1CC1)C C(CCCCCC(=O)NC)n1cc(-c2c(C)nn(C)c2)nn1.C(C(=O)O)SC(F)F N1(C(C(CC)C#N)=O)CCCC2(NC(C3CC4CC4C3)=O)CCCC12 c1(C2CCN(C(C3N(C(C)=O)CC3)=O)C2)ccc(SCCC(=O)OCC)cc1 C12(C(N(CCCNC(=O)Cn3cccnc3=O)C3CC3)=O)CCCN1CC(O)C2 C1(C(=O)NCCN(CCC)CC)(CNC(=O)Cc2cc(C)cs2)CCCO1 N1(C(c2cn(CC(C)C)nc2)=O)CCC(CN(C(=O)C=C2CC2)C)CC1 C#CCC(C(=O)N(CCCOC)CCO)CCNC(=O)COc1cnn(C)c1 c1(OCC(CNC(=O)NC2CC(CCOC)C2)O)ccc(Cl)cc1F Cc1nc(CCC(=O)NC2CC(NC(=O)CCc3csc(C(C)C)n3)C2)cs1 C1(C)(CNC(c2ccc(C)cc2)=O)CCCN(C(=O)CC2CSC2)C1 CC1=CCC(C(=O)N(C2CCCC2)CCNC(c2cc(Br)n[nH]2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)N1CC2(OCC(NC(C3CC(C)OC3)=O)C2)C1 Cc1cc(N2CCN(CC(=O)NCc3cc(F)ccc3Cl)CC2)nc(CC2CC2)n1 c1(OC)cc(C)c(C(N2CCOCC2CCNC(=O)CN=S(C)(C)=O)=O)cn1 c1(C(=O)NC(CC)CNC(=O)C(C)c2cncs2)cc(C)ccc1S(N)(=O)=O N1(C(Cc2nc(CC)sc2)=O)CCC(C2CN(C(=O)C(F)n3ccnc3)C2)CC1 C(=O)(C1=CCCCCC1)N1C(CNC(=O)Cn2nc(Cl)ccc2=O)CC(O)C1 C1(NC(c2c(CNC(CNC(CCC)=O)=O)ccs2)=O)CC(CO)C2CC12 CC(N=c1[nH]c(=NCCc2cn[nH]c2)c2c(ncn2C)[nH]1)c1c(F)cccc1Br N1(C(C(C)(C)O)=O)CC2CCCC(CNC(C3CC34CCCCC4)=O)C2C1 C(=O)(CCCCN=[N+]=[N-])N1CCC(C(C(N2CC(CC(=O)OCC)C2)=O)C)CC1 C(=O)(C(F)CC(C)(C)NC(=O)CCS(C)(=O)=O)N1CC(C(N(C)C)=O)C1 C12(C(C)C)COC(CNC(=O)Cc3ccon3)(C1)C2.C1(C(=O)NC)CCCCC1 c1(C(N2C3C(C(N4CC(C(C)C)OCC4)=O)C(C3)C2)=O)cc(Cl)c(Cl)nc1Cl C=CC(C)(O)CCCC(C)C(=O)N1CCC(CCNC(=O)C(F)=CC2CC2)CC1 C1(NC(C(CC)N(C)C)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C)nc1 c1(C(=O)NCC2C3CN(C(C4(C)CC4(F)F)=O)CC32)[nH]nc2ncnc(O)c12 C(CNC(=O)Cc1nocc1C)(CC(=O)NC(c1csc(C)n1)C)OC CC1C(C(=O)N2CCC(C(C)C(=O)N(C)CC3(O)CCOC3)C2)=NOC1C N1(C(c2ncn(C)c2)=O)CC2(CCN(C(=O)C(c3ccc(Cl)cc3F)O)CC2)C1 N1(C(C=C(C)I)=O)CC2CCN(C(=O)CCc3ccccc3)C2C1 Cc1sc(=NC2CCOC3(CCN(C(=O)Nc4ccccc4)CC3)C2)[nH]c1Cl N1(C(C(CC#C)C2CC2)=O)CCN(C(c2cc3occc3[nH]2)=O)CC1C1CCC1 c1(C(=O)NC2C(CNC(C(CSC)C)=O)CCCC2)ncnc2c1cnn2C Cc1cn2c(n1)C(C)CC(NC(=O)NCC1CC(=O)NC(=O)C1)C2 c1(C(C(=O)NCC=C)N(c2ccc(OC)cc2)C)ccc(CC)nc1C C1(OC)CC(C(=O)O)CCN(C(=O)CSC(F)F)C1.c12ccncc1C(=O)N2 Cc1cc(C(=O)NCC2(O)CCN(C(=O)C=Cc3cn(C)cn3)C2)c(C)s1 c1(C(=O)NC2CCN(C(CCCOCCC)=O)CC2F)nnc2n1CCCC2 C1(C(=O)NCC2(OC)CN(C(Cc3ccc(OC)s3)=O)C2)COCC(C)(C)O1 c1(C(=O)NC2C(NC(CC=CC=C)=O)C2)cc(N2CCNC2=O)ccc1F Cc1ccc(C(=O)NC2CS(=O)(=O)CC2NC(=O)CCc2ncco2)cc1Cl c1(C2(NC(=O)NC3CC3c3ccc(Br)s3)CCC2)cccc(OC(F)F)c1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCC2(CC1)C(=O)N2CC.C1(Br)(SCC)CC1 Cc1nc2cccc(C(=O)NCCC(C)NC(c3ccoc3C(C)C)=O)c2[nH]1 N1(C(C2C(C)(C)C2)=O)CC(CNC(=O)CNc2ccccc2C(N)=O)CC1(C)C CCCC(C(=O)N1CCN(C(c2c[nH]c(C#N)c2C)=O)CC1CC(F)F)C(C)C C(=O)(C(=O)C(C)C)N1CC(C(F)(F)CO)(NC(C=CC=CC)=O)C1 CC1CN(C(C2(c3cccnc3)CC2)=O)CC1NC(c1nc(Cl)cs1)=O C(=O)(CCS(C)(=O)=O)N(CCN(C)CC1CCCN1Cc1csc(Br)c1)C N1(C(CCCCC=C)=O)CCC2(CCCN(C(=O)CC3CCCN3CC)C2)C1 C1(CC)CCCN(CC(=O)NC2(CN(C)C(C3C(Cl)(Cl)C34CC4)=O)CC2)C1 N1(C(C(c2ccccc2)NC(CC(C)(F)F)=O)=O)CCC(O)(CO)CC1 S(=O)(=O)(c1ccc(NC2(C)CC(F)(F)C2)c(F)c1)N(C(c1ccncc1)C)C1CC1 CCC1=C(C(=O)NCC(C)CNC(c2[nH]ccc2C(=O)OC)=O)CCCO1 c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ccc(Cl)cc1Br C1(NC(CC2CC(C)C2)=O)CCCN(C(c2ccsc2)=O)C1C C1(F)(C(=O)NCC(C2CCN(C(c3ncsc3C(C)C)=O)CC2)F)CCCCCC1 c1(C2C(C(=O)NC3CCN(CCOC)C3)C2)nn(C)c2ccccc12 N1(CC(=O)NCCOCCN(C)C(c2csc(C(N)=O)c2)=O)C(=O)CN(C)C1=O Cc1oncc1S(=O)(=O)N1CCC=C(C(=O)Nc2nc(C#N)cs2)C1 C12(C(=O)Nc3cccc(-c4ccc(C(C)C)cc4)n3)C3C4C1C1C2C3C41C(=O)O c1(OC)cc(O)c(C(N2CCOC(C)(CNC(=O)C3CC3)C2)=O)cc1F c1(C(N2CC(NC(=O)C=Cc3ccoc3)CC(C)C2)=O)cnn2ccccc12 c1(C(N(CCOC)CCNC(=O)Cc2csc(C)c2)=O)ccc(Br)cn1 c1(CN2CCC(NC(c3ccc(C(=O)OC)cc3C)=O)C2)ccc2cc[nH]c2n1 c1(C(=O)NCC2C(NC(CC3C(C)(C)C3)=O)C2)ccc(=N)[nH]c1 CCCC(CCCNC(c1cnc(O)cc1C)=O)NC(=O)Cc1c[nH]nc1O c1(CCC)n[nH]cc1C(=O)NC1CC1NC(c1coc(C2CCCCC2)n1)=O C1(S(C)(=O)=O)(C(=O)NCC(C)CNC(c2cnc(Cl)s2)=O)COC(=O)C1 N1(C(Cc2cnc(C)s2)=O)CCC(F)(C(=O)NCC2(O)CCCOC2)C1 C(=O)(CC(O)C(C)C)N(C1CCCCC1)CCNC(c1c(C#C)c[nH]n1)=O c1(C(NNC(COc2cccc(SC)n2)=O)=O)ccc2c(c1)OCO2 Cc1ccc2scc(CC(N3CCC(NC(=O)C=CC4CC4)C(F)C3)=O)c2c1 c1(C(N2CCN(C(C3CCC(F)(F)C3)=O)C3CC23)=O)cc2cccc(Br)c2[nH]1 C1(NC(COCC(C)(C)C)=O)CCC(NC(c2cn(C3CC3)cn2)=O)CC1 C(C)(CC(F)(F)F)N(C1C2(CCCCC2)NC1=O)C.CCC(C)(C)OC C12CCCN(C1=O)CC(=O)N2.c1(C(CC=C)OC)cn(C2CC2)nn1 C1(CNC(C2C(OCC)CC2)=O)CC2CC2N1C(c1ccnn1C1CC1)=O C=C(C)CC(C)C(=O)N1CCC(C(C)NC(c2cscc2SC)=O)C1 Cc1nc([N+](=O)[O-])cn1CCC(=O)NCC1CC1NC(C1C2CCCCCC12)=O C1(CNC(C(C)S(C)(=O)=O)=O)CC12CCN(C(=O)C=Cc1ccccc1)CC2 C1(N(C(=O)CCCc2ncco2)C)CCC(NC(=O)C(C)(C)n2cc(Cl)cn2)CC1 C(=O)(CCCCn1cc(-c2cnc(-c3cccs3)s2)nn1)N(C)CCOOCC.N C1(COC(c2ccc(OC3COC3)nc2)=O)OCC2CC(=O)C1C2 c1(NC(CCC)=O)ccc(COC)nc1C.N12CC=CC1(COC)C2=O c1(C(=O)OC(CC(=O)OC)C)cccnc1C(F)(F)F CCC(N=c1cnc(C(=O)OC(C)=O)c[nH]1)C1CCCOC1 c1(OCC)cc(Br)ccc1C(N1CC(C(=O)Nc2cccnc2Cl)C1)=O C(C(C)(C)C#CC(=O)NC(CCO)c1ccco1)NC(C1CCN(C)C1=O)=O c1(C(N(C)CC2COCCN2C(C2COCCO2)=O)=O)cc2cn[nH]c2cn1 C1(C(=O)NCC2(CO)CCCO2)CCCCC1NC(C1CCCC1O)=O c1(C(N2CC(C)(NC(c3c(C(C)C)ncs3)=O)C2)=O)cc(F)cc2nc[nH]c12 c1(C(=O)NC2C3(CC(NC(C(CC=C)CC)=O)C3)C2)cn2c(Br)cnc2s1 N(C1CCc2ccc(Cl)cc21)CCCCCC(=O)NC1CCC(=O)NC1 N1(C(c2n[nH]c(C)c2C)=O)CC(NC(c2cccc(Cl)c2N)=O)CC(O)C1 c1(CC)onc(C)c1C(N1CC(N(C)C(c2ccn(C(C)(C)C)c2)=O)C1)=O C12(CNC(C(C)(F)F)=O)CCC(CC1)CN2C(c1c(Cl)cccc1Br)=O Cc1noc2ccc(C(=O)NC3(C)CCN(C(=O)C(=C4CCCCC4)F)C3)cc12 C(=O)(C(O)CC(F)F)N(c1ccc(Cl)cc1Oc1ccccc1)C C1(O)(CNC(C2(CC)CCC2)=O)CCCN(C(C2CN(C)C(=O)CCO2)=O)CC1 c1(CN2CC3(CC(NC(C4(F)CCCNC4)=O)C3)C2)cc(F)c(F)cc1Cl C1(CN)CC(O)CN1C(c1ccc(N2CCCC2=O)cc1)=O N1(C(CC2CCC(C)CC2)=O)CCCC12CCCN(C(=O)C(N)=O)C2 C1(CNC(CCC=CC)=O)C2CN(C(C3(CCC)CCC3)=O)CC12 c1(C(=O)NCc2cc(C(N3C(COC)CCCC3)=O)on2)cnccc1C#N C1(C(=O)NC)CCOCC12CCC2.C12CC(C1)C(=O)N2.C12(CC1)CC2.CCOC N1(c2c(C#N)cncc2)CCCC12CCN(C(=O)CCC1CCC1)CC2 C=CC(CCC)CC(=O)NC1(C(N2CC(O)(CCC)C2)=O)CC1(C)C C1(C)(C(C)NC(C2(CNC(CN(C(COC)=O)C)=O)CC2)=O)CCCO1 C1(C(=O)NC)CCN(C(C2(C)CN(C(=O)CNC=O)C2)=O)C1 c1(CCC(=O)NC2CCC2CNC(=O)Cc2ncoc2C2CC2)ccc(Cl)s1 N1(C(c2c(C)csc2)=O)CCCN(C(C2CCCC(C(N)=O)C2)=O)CCC1 C12(n3cc(CC(C)(C)CO)nn3)CC(NC(=O)Cc3ccsc3)(CCO1)C2 C(=O)(C(=O)C(C)(C)C)NC1(C(=O)NC(c2cnccn2)C)CC(F)C1 c1(OC)cccc2cc(C(C)NCC(C)(C(=O)O)n3cc(Br)cn3)oc12 N1(C(C2N(CC)CCC2)=O)CC(F)(F)CC1C(=O)N(C1CCCN1)C1CC1 C(=O)(C1=CCCOC1)N1CC2C(CNC(c3ccnc(C(F)(F)F)n3)=O)(C2)C1 c1(CC(=O)NC2CCCC(N(C(=O)CC3CC3)C)C2)cccc(C#N)c1 C(C)(CC(=O)NCCN(C1CCC1)C)N(C(C(C1CCOCC1)C)=O)C c1(NC(CC2(C(=O)OC)CCNC2=O)=O)cccc([N+](=O)[O-])c1Br C1(CC(=O)NCC(CC=C)NC(c2ccc(Cl)cc2O)=O)COCC(C)(C)O1 c1(C(=O)NC2CCC(CNC(CC3CC(CC)C3)=O)C2)cccn2c(C)cnc12 c1(C(=O)NC2C(CNC(CCCOC(C)(C)C)=O)CC2)cn2c(n1)SCC2 Cc1ccc(O)cc1C(N1CCC(C(C)C(=O)N(CCS(N)(=O)=O)C)CC1)=O c1(C(=O)NCC2CCN(C(CC3C(C)OCC3)=O)C2)cnn(C)c1C(F)F Cn1nc(C(F)(F)F)cc1NC(C1CCC(CNCc2ncccn2)CC1)=O c1(C(CO)C)cc(F)cc(F)c1.C12CCN(C1=O)C(C)O2.c1(C)ccccc1 C1(NC(C2(C)COC2)=O)CCC2(CC1)CN(C(=O)Cc1ccc(Cl)s1)CCO2 C1(C(=O)NCC2C(NC(c3n[nH]c(C4CC4)n3)=O)CCCC2)CC12CCSCC2 N1(C(C(N)=O)=O)CCC2(CC1)OCCC2NC(=O)CCCc1ccc(Cl)cc1 c1(NCCCOC(C)C)cc(NC(=O)CN(C2CCCC2)C)ncn1 C1(CNC(=O)Nc2cc(O)n[nH]2)Cc2ccc(Br)cc2C1 N1(C(C(C)c2ccco2)=O)CCN(C(c2cn3ccnc3s2)=O)CC(O)C1 c1(C(=O)NC(C(C)NC(c2n(CCC)ncc2)=O)C)ccc(C2CC2)cc1F Cc1c(C(N2CCN(C3CCCN(C(C4CC45CC5)=O)C3)C(=O)C2)=O)cncc1Cl C12(NC(C)=O)CCC(CN(C(c3c[nH]nc3-c3ccc(F)cc3)=O)C1)C2 C1(C(C)NC(C=COCC)=O)CCCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)C1 C(CN=c1[nH]c(C2CC2)nc(C2CC2)c1C)N(CCC)C(C1(CC)CCC1)=O.C N1(C(c2cc(CC)sn2)=O)CC(F)(F)CC1C.C12CC3(C1)CC3C(=O)N2 CCCCCCC(C)C(=O)NC(C)CNC(=O)CC(C)CC(=O)OC c1(C(=O)NC(C(=O)NCCCOC)CCN(C)C)ccc2ncccc2c1F Cc1cccnc1C(=O)NC1CCCN(C(=O)CC2(C)CCOC2)C1 C1(C(=O)NC(CN(C(=O)C=C2CCC2)C)(C)C)CS(=O)(=O)CCO1 CCC(CC)CCC(=O)NCC(CC1CCCC1)C(=O)NC(C1CCN(C)C1)C C1(NC(c2cc(C(CC)CC)no2)=O)CCN(C(=O)CNC(=O)CSC)C12CC2 c1(SC)nc2ncnc(N3CCCC(NC(=O)C(C)CSC(F)(F)F)C3)c2s1 C1(C(=O)NC2CN(C3CN(C(CCSC)=O)C3)C(=O)C2)CCOCC12CCCC2 C(=O)(CC(C)(C(F)(F)F)n1cc(-c2ccc(F)cc2)nn1)NCC(C(C)C)C(=O)O C1(CNC(c2ccc(SC)cc2)=O)CCN(C(=O)CCCc2cccs2)CC1C c1(CN2CCC(CNC(Cc3ccc(C)cc3)=O)C2)ccc(N(C)C)c(Br)c1 c1(OC)cccc(CSCC(=O)NC2(C)COC2)c1OC c1(C(N2C3(CN(C(C(C)(C)C(F)F)=O)C3)CC2)=O)cccc(O)c1[N+](=O)[O-] C1(C2CCNCC2)(c2nc(C(CCCC(C)C)C)on2)CCOCC1 C12(C(=O)NC(C(C)SC)C)CCC(CC1NC(=O)CC1(C)CC1)C2 N1(C(c2occ(C)c2C)=O)CC2CC3CC2C1C3NC(c1ncc(F)cc1F)=O c1(OC)ccc2c(c1)CCCC2C(=O)N1C2CCC1C(CNC(=O)C(C)(C)C)C2 c1(C(N2CCCC(N(C(C3C(C=C)C3)=O)CC)C2)=O)cc(O)nc(O)c1 c1(CCC=C=C)nc(C2Cc3ccccc32)nn1C(C)C(C)C N1(C(CCOC)=O)CCN(CCOCCCNC(C2(C#C)CCCC2)=O)C(=O)C1 N1(C(c2ccccc2N2CCCOCC2)=O)CCNCC1CCO CN(C(=O)c1ccccn1)n1cc([N+](=O)[O-])cn1 C1(C2N(C(C=C(C)Cl)=O)CCC2)CCCCN1C(=O)CCOc1ccccc1F CC1CCN(C(c2cnn(CC(F)F)c2)=O)CCN1C(C1CCN(C)S1(=O)=O)=O N1(C(c2c(CC)n(CC)nc2)=O)CCC(C)C(N(C(=O)CN2CC(F)(F)C2)C)C1 CCC(CC(=O)N(CC(C)NC(=O)CCNC(=O)CC(C)C)CC)C(C)C CCC(CC)C(C)C(=O)NCC1CC2CCC1N(C(=O)C(C)(C)CO)C2 c1(C(=O)NC(C)CCNC(=O)C(C)NC(c2ccco2)=O)ccn2c1CCC2 CCCCC(F)(F)C(=O)N1CCC(NC(c2ccnn2COC)=O)C(CC)C1 N12CCC3CC3(CC1)C2=O.N1(CC2CN(C=O)C2)CCC(n2ccnn2)C1.CCSCCl Cc1cc(CNc2cccc(C(=O)NOC3CCC3)c2)c(C)n1-c1ccccc1 C1(C(=O)NCC(c2cccc(OC)c2)NC(CCCCC)=O)CNC(=O)CC1C c1(C(N(CC(C)N(C(=O)C=CI)C)C)=O)ccsc1C(F)F CC(C)C(F)(F)CC(=O)NC1CCN(C(c2ccc(C(C)(C)C)cc2)=O)C12CC2 C(=O)(C(C)(C)CC(C)C)NC(CNC(c1c(C)ccnc1C)=O)CC(C)C C1(C(N(CCN(C)C(c2n[nH]c(O)n2)=O)C)=O)CCC2(CC1)CC2 c1(CNC(C(C2CCC2)NC(CCOCCOC)=O)=O)ccc(Cl)cn1 C1(NC(CCCCC)=O)CC2CC1CN2C(c1cn(C)nc1-c1ccncc1)=O c1(C(=O)NC(CC(C)NC(c2cc(C)c(C)o2)=O)C)ccc2nc(C)n(C)c2c1 C1(C(N2C(C(=O)NCC(C)OC)CCCC2)=O)CC2CCC(C1)O2 C1(NCC2C(C(=O)OCC(N(C3CCOC3=O)C)=O)C2(C)C)CCC(=O)N1 C#CCCC(C(=O)N1CCCC(C)(N(C)C)C1)NC(=O)CCc1ccnn1C O=C(CC(CC1CC1)NC(C1CCCCC1F)=O)NC1(C2CCCCO2)CC1 c1(C(=O)NC(c2cccnc2)C(=O)N(CC)CC2COCCO2)ccncc1Cl c1(C(N2CCCC(CO)C2)=O)ccc(N)cc1Cl.c12cc(on1)CN(C)C2=O C(C(CC(C)C)NC(C1CC=CCC1C)=O)NC(C(CC1CC1)OC)=O C1(C(=O)NC2(C(N(CCC#C)CC)=O)CCSC2)C(C#N)C1(C)C c1(C(=O)NCC(C)NC(C2C(COC)C2)=O)ncc(N)cc1C c1(CCNC(N2CC3=CC(=O)SC3CC2)=O)ccc2ccccc2n1 N1(C(C(C)Oc2cccnc2)=O)CCC(NC(c2nnn(C(C)(C)C)n2)=O)C1C C1(NC(C2=NOC(C)(C)C2)=O)CCOC2(CCN(C(=O)C=CC3CCC3)CC2)C1 c1(C(N(C)CC2C3CN(C(C4CCC4)=O)CC23)=O)ccc2c(n1)NCC(=O)N2 CC1CCC(CC(=O)NCC2CN(C(=O)COC3CCOCC3)C2)C1 CC(C(C)(C)C)=CC(=O)NCC1OCCC1C(=O)NCCCCN(C)C C(=O)(C(F)C(C)(C)O)N(C(C)CN(C(=O)CSCc1cscn1)C)C C(=O)(C(C)(F)CC1CC1)NCCC(CNC(C(C)C)=O)O C#Cc1cnc(C(=O)NCCCCC(N2CCSC3CCCC23)=O)c(C)c1 c1(OC)cc(C(C)(C)CNC(=O)C(=O)NCc2cc(N)ccn2)ccc1Br n1(CC(C(=O)N(CC(C)(C)NC(CC(COC)C)=O)C)(C)O)ccc(C)cc1=O c1(C(N2CC(CNC(C(C)(F)F)=O)OCCC2)=O)nc2cccnc2s1 C1(NC(c2c(C)con2)=O)CCN(C(C2CC(=C3CC3)C2)=O)CC1O N1CC2CC1CN2C(c1nc(C2CC2)no1)CO.Cn1cc(OCC(=O)N)cn1 N1(C(C(CC)CCOC)=O)CCC2CN(C(c3cccc4c[nH]nc34)=O)CC12 N1(C(CCCCCC)C(=O)NC(C)C)CCC(C2CC(O)C2)CC1 C12(Cc3cn(CC(=O)OC)nn3)CCC(CC1)N2C(=O)CN1CCS(=O)(=O)CC1 Cc1noc(CNC(C2(C)CC(O)C2)=O)n1 c1(CC)cccc(C(=O)NCCC2CCN(C(C3CC(=O)N(CC)C3)=O)C2)n1 CS(=O)(=O)CCCCNC(C1(CNC(c2ccc(F)c(F)c2)=O)CC1)=O c1(CC(=O)N(C(C)CNC(=O)CS(=O)CC)CC)ccc(C)cc1Cl C=CC1(C(=O)NCCC(C)C(=O)OC)CCN(C(=O)C(C)OC(C)=O)C1 c1(C(N(C(C)CN(C(=O)CC(C)c2ccncc2)C)C)=O)cc(O)nn1C c1(C(N2CCOC(C3(O)CCCC3)C2)=O)cccc2ccsc12 N1(C(=O)Cc2cc[nH]n2)CCC2(CCCN2C(=O)CCCC2CC2)C1 C(CO)(C(C)N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC3CCCC3)cc2s1)SC c1(C(N(CC)Cc2cn(-c3ccc(C)c(Cl)c3)nn2)=O)cncc2ccccc12 C1(C(N(CCCNC(=O)C(F)(F)CC2CC2)CC)=O)COCCC1(F)F N1(C(c2n(CC)ncn2)=O)CC2(CCN(C(=O)C(C)=C(C)C)CC2)C1C(C)C C12CCN(CC1O)C(=O)N2C.c1(N(C2CCC2)C(=O)C2CC2)cc(Br)ccc1F N1(C(C=CC=CC)=O)CCC(C(=O)NC2CC2C)C1C C=CC(C)(C)CC(=O)NC(C(C)NC(=O)C=Cc1csc(C)n1)C(C)C C(=O)(C1=CC2CC(C1)CC2O)NCC1(OC)CCC1.c12nc(cs1)CC(=O)NC2 N1(C(=O)CC2CC3CC3C2)CC2(CCN(C(C3(C(N(C)C)=O)CC3)=O)C2)C1 Cc1nn(-c2ccccc2)c(Cl)c1C(=O)NN1C(C)C(C)CC1.c1(C)ccccc1 c1(C(=O)NC2(C3N(C(CCOC(C)C)=O)CCC3)CC2)ccc2cc[nH]c2n1 Cc1c(C(=O)NCCOC2CCN(C(=O)C(C)C3CC3)C2)sc2cccc(F)c12 C1(N(C(=O)CCn2cccc2)C)CCN(C(=O)CC2CCCOC2)CC1 C1(OCCNC(C(C)SCCCC)=O)CCN(C(=O)COCC2CC=CC2)C1 C(=O)(CC1=NN(C)C(=O)C1)NCCNC(c1c(Br)ccc(C)c1)=O N1(C(Cc2c(C)nsc2)=O)CC(F)CC1CNC(C1CCC(=O)NC1)=O c1(C(=O)NCC(C)(CNC(=O)C(C2CCOC2)OC)OC)cccc(O)c1 c1(C(N(C(C)C)CCN(C)C(C23CCC(C2)C3)=O)=O)cccc(C(C)(C)C)c1 Cc1c(NCc2ncc(F)cc2F)ncnc1NC1CCN(C2CC2)CC1 C1(NC(CC2C(C)C2(F)F)=O)CCN(C(c2ncccc2N)=O)CC1(C)C C=C(C)CCCC(=O)N1CC(C2CN(C(=O)C(C3CCOCC3)C)CCO2)C1 N1(C(CCC2CCCN(C)C2)=O)CCC2(NC(C3CC4CCCC34)=O)CCCC12 Nc1cc(C(=O)NC2CCC(CCNC(=O)CC3CCC3)C2)cc(O)c1Cl Cc1cscc1C(N1CCC(N(C(=O)CC2CC(F)(F)C2)CCO)C1)=O N1(C(C(Cn2cncn2)NC(CN(C)CC)=O)=O)CC(C2(C)CC2)C1 c1(CCC)nc(C(=O)NCC2(CNC(=O)COc3ccccc3)CCC2)co1 N1(C(Cc2cccc(C)c2C)=O)CCC(NC(C2(CCO)CC2)=O)C(CO)CC1 Cc1occc1CC(=O)NCC1CCCN1C(=O)CC1(N2CCCC2)COC1 C(C(CC(F)(F)F)NC(C1(C)CC(C(F)(F)F)C1)=O)NC(C(CC)SC)=O N1(C(c2cc(C)sn2)=O)CCC(C(=O)NCC2C=CCOC2)CC1 c12ccc(cc1Cl)NC(=O)C1C(C1)C(=O)N2.C(C)(C)(C)OC(CCOC)=O N1(C(C2CC(SC)C2)=O)C2CCC1CC(CCNC(=O)C=CC1CCOC1)C2 c1(-c2onc(COC(c3ccc(CCC)[nH]3)=O)n2)ccccc1Cl N#Cc1ccc(S(=O)(=O)NC2CCCc3cc(N)ccc32)cc1 C1(NC(CCSC)=O)CC(O)CN(C(=O)COc2c(F)cccc2F)C1 CP(C)(=O)C1CCCC=C1C(=O)N1CC(F)CC1CNC(C1CC2CCC1O2)=O C1(c2cn(CCN(C(=O)CSc3cccc(C)c3)CC)nn2)CC2CCC1CC2 N12CCC(CC1)NC(=O)C2C.c1(C(N2CC(F)(F)C2)=O)cc(C(N)=O)c[nH]1 c1(C(N(C2CC(NC(=O)C(F)=C3CCCC3)C2)C)=O)cc(-c2ccns2)on1 C12(C(=O)NCC3CC(OC)CN3C(=O)CN3CCCC3=O)CCC(N=[N+]=[N-])C1C2 C(=O)(CCCC1CCOCC1)NC(C1CN(C(=O)C(C)N2CCC2)C1)C c1(NC(C2(C)N(C(c3nn(CC)c(C)c3)=O)CC2)=O)ccc2nc(O)oc2c1 N1(C(C(CC(=C)C)NC(C)=O)=O)CCC(C2CCN(C(C3C(C)C3C)=O)CC2)C1 C(C(=O)NCCC1CCN(C(C2CC(OC)C2)=O)C1)(C(C)C)NC(C(C)C)=O C1(CN2CC(C)C(c3ccc(Br)cc3)C2)CC2COCCC2O1 C1(C(N2C(CC(=O)NC)CC2)=O)CCCN(C(C2CC(=O)OC2(C)C)=O)CC1 N1(C(CCCC=C)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CC12 c1(C(N2C3C(NC(c4ccc(Cl)cc4F)=O)C(C3)C2)=O)ccc2n[nH]cc2n1 c1(-c2cc(CN(C(C)CNC(c3cscn3)=O)C)no2)ccc(F)cc1 c1(C(=O)NCC(C2CC2)NC(C2C(C#C)C2)=O)c(Cl)c2ccccc2n1C C1(CC)CN(C(c2cn(C)nc2C)=O)CCN1C(=O)Cc1cccc(O)c1 N1(C(c2cncc(C)c2)C(=O)NC2CCC2)CC(C)N(S(C)(=O)=O)C(C)C1 c1(NC(N2C(C(=O)Nc3c(C)c(O)cs3)CC(F)C2)=O)n[nH]c2cccnc12 c1(OC(C(=O)NC(CN(C(CCC)=O)CCOC)C)C)ccc(Cl)c(C)c1 c1(C(=O)NC2(CCOC)CCN(C(c3cncs3)=O)C2)nccc2ccn(C)c12 Cn1cc(C(=O)NCC2CC2CNC(=O)Cc2ccn(-c3ccccc3)n2)cn1 N1(CCCOCC)CCCC(C)(NC(C2(C)CNC(=O)C2)=O)C1 C1(N(C(c2ncc(C)s2)=O)C)CCCN(C(c2n[nH]c(C3CC3)c2C)=O)C1 CC1CCCCN(C(c2ccncc2-c2ccccc2Cc2ccccc2)=O)C1 c1(C(=O)NC2CCN(C(C3(C)CCCCO3)=O)C2)cc(N)ccc1Cl Cc1ccc(NC(=O)CC2CCCN2C(c2nccn3ccnc23)=O)c(C)c1C c1(C(C)NC2CCC(n3cc(COC)nn3)CC2)cn2ccccc2n1 c1(-c2nc(SCc3cn(C(C)C)nc3)on2)ccccc1C(F)(F)F CC(C)C(O)C(C)C(=O)NCCc1nc(C(=O)N(C)C(C)C2CC2)co1 c1(CN(c2nc(OC)c(F)cn2)C2C3CCC2CNC3)cc(F)c(F)cc1C c1(CN(C(=O)C(C2CC3CCC2C3)(F)F)C2CC2)cc2cccc(C(=O)O)c2s1 c1(NC(C)=O)c(C)cc(C(N2CCCCC2C2CCNCC2)=O)cc1C N1(C(CC(CC)C2CC2)=O)CCOC(C)(CNC(=O)C(c2cccn2C)=O)C1 C1(F)(C(=O)NC(C)CCO)CCCN(C(C2CCOC(C)(C)C2)=O)C1 c1(C(=O)NCC(=C)CCNC(=O)C(C)CCOC)cc(C#N)ccc1Cl CC(C)CC(CN=c1cc(Cl)nc[nH]1)NC(=O)C(C)(O)C1CCC1 C1(COC)CC(CNC(C2CCCCS2)=O)N(C(C2CCC(C(N)=O)CC2)=O)C1 N1(C(c2cnn(C)c2Cl)=O)CC2CCC(Nc3ncn(C)c(=O)c3Br)C2C1 C1(C(N2CC(CC)C(C(N3CCCC3)=O)C2)=O)CCc2n[nH]cc2C1.C1(=O)CN1 C1(OCC(=O)Nc2ccccc2OC(F)F)CCCc2ccccc2C1 CCCC(C(=O)NCC1C2CCCC12)NC(c1cc(C(C)C)[nH]n1)=O c1(C2C(C(=O)NC(CCCOC)c3cccnc3)C2)ccncc1F c1(C(N2CC3CC(NC(C4(C)CCCCO4)=O)C3C2)=O)cc(F)cc(F)c1O N1(C(C(C=CC)O)=O)CCC2(CCC(CNC(=O)C(C)C3CCOC3)CC2)CC1 CC1=C(C(=O)O)CCN(C(C2CCCC(C(=O)Nc3ccccc3)C2)=O)C1 CCC(C)C(O)C(C)C(=O)N1CCN(C(=O)C(F)F)CC1Cc1ccccc1 Cc1ccnn1C(C)C(=O)NC1(C(=O)NC(C)CCOC)CC1 C1(C=C)(C(=O)NCCOCCC=C)CCN(C(C2CCCC(F)C2)=O)CC1 O=C1CCOC(C(=O)NCC=CCC(N2CCC(F)(C(N)=O)C2)=O)C1 C1(NC(c2c(CC)c[nH]n2)=O)CN(C(c2nccn3cnnc23)=O)CC12CCC2 C1(NC(CC2(CC)CCC2)=O)CCOCC1C(=O)N(CCn1cncn1)CC N1(C(CNC(CC(C)C)=O)=O)CCC(O)(C(=O)NC(Cc2ccccc2)CO)C1 C1(O)(C(C(=O)OCC)(F)F)CCN(c2nnnn2CC2CCCO2)CC1 C(=O)(C(C#N)C(C)C)NCC(CCCC)NC(=O)CN(C)C(C)=O C1(CC(=O)NC(c2nccs2)CC)CC2CNCC2O1 C#CC1CN(C(=O)C(C)(C)C2CCN(C(=O)CC(C)F)C2)CCO1 S(=O)(=O)(c1ccc(C)cc1)N1C(C(=O)NCCNC(CCOC)=O)CCC1 c1(C(C)(C)C)cccc(CNC(c2coc(CNC(=O)C(N)=O)n2)=O)c1 C(=O)(CC(C)CC(=O)NCC1CCCN(C(=O)CC2CCC2C)C1)OC c12ccc(nc1)NC2.c1(C(N(CC=C)CC=C)=O)c[nH]nc1C1CCC1 Cc1cnccc1C=CC(=O)NCCC(O)CNC(c1ccc(Br)cn1)=O C(=O)(C(CO)C(C)(C)C)NC1C=CC(CNC(c2cc(OC)ns2)=O)C1 C(=O)(CCN(C(=O)CCC1OCCO1)CCO)NC(COCC)C C12(NC(c3cc(C)sn3)=O)CN(C(c3ccc(CO)o3)=O)CC1CS(=O)(=O)C2 c1(C(=O)OC)cc2oc(C(=O)NC(CNC(=O)C(C)C(C)O)CC(C)C)cc2[nH]1 C1(N(C(=O)CCC(=O)NC(C)(C)C)C)CCCC(NC(C2CC2(F)F)=O)C1 Cc1ncc2c(n1)CCC(C(N1CCC(C)(NC(C3CN(C(C)C)C3)=O)C1)=O)C2 c1(C(N2CC(NC(C3ON=C(C(C)C)C3)=O)C2)=O)cnc(C(F)(F)F)c(Cl)c1 N1(C(c2n(CC)nc(C3CC3)c2)=O)CCC2CN(C(c3cnsc3)=O)CC2CC1 N1(C(C23CN(C(=O)CC4(O)CCCC4)C(CC2)CC3)=O)CCC2(CCCOC2)C1 C12(C(=O)NCCC3(O)CN(C(c4c(C)ccnc4)=O)C3)CCCCC1CCC2 N1(C(CN2CCC(C)CC2)=O)CCCN(C(=O)C(O)CC(F)F)CC1 c1(OC)ccc(-c2ccc(CN(C)Cc3cccnn3)s2)cn1 CC(C(=O)NC1(CN(C)C(c2cc(F)ccc2O)=O)CC1)C(F)(F)F C#CC1CN(C(=O)C(C(C)OC)N(C)C)CCN1C(c1ccc(Cl)cc1C)=O C1(NC(C)=O)CN(CC(O)COCC(C)C)CC1(C)C CC(C(=O)NCC1CCOC1C(=O)NC(C)(C)CCCO)C(F)(F)F C(=O)(CC(C)(C)CC(F)F)N1CCC(C(=O)NC(C)CC(F)F)CC1 CC1(C)CC(C(=O)NCCCC2CCC2)CCN1C(C1CC2(CCC2=O)C1)=O Cc1ccc(C(=O)NCC(C)(C)OCCCNC(=O)Cc2nc(=N)[nH][nH]2)n1C CCC(CC(F)(F)F)C(=O)NC(C)C(CO)NC(=O)C(c1ccccc1)=O C1(O)(c2scc(CC(N3C(CNC(C=CCC)=O)CC3)=O)n2)CCOCC1 Cc1c(C(=O)NCC(C)CNC(c2cc(O)nn2C)=O)nnn1C1CCOC1 C=CCCCCC(=O)N1CCC(N(C(=O)Cc2nc(C(C)C)c(C)s2)C)C1 C#Cc1cc(C(=O)NC2CCN(C(=O)C(F)F)C(C3CC3)C2)cc(Br)c1 C#CCCC(C(=O)NC1CCS(=O)(=O)C1)NC(c1cc(F)cnc1O)=O c1(C(=O)NC2CC3(CC(NC(C4CCC(OC)C4)=O)C3)C2)cc(C)c(C)cc1C N12CCCC(C1)OC1CCN(C1)C2=O.C1(CCOC)(CO)CC1 C(=O)(C1CCCc2c1ncn2C)NCC1CC(NC(c2ccn(COC)n2)=O)C1 C1(NC(COCCC=C)=O)CN(C(c2cnc(NC)cn2)=O)CCC12CCC2 c1(OCC(=O)NCCCNC(CCC2CCC(C)O2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCCN(c2cc(C(C)=O)ncn2)CCC)ccc(C=NOC)cc1 c1(N)ccccc1Cl.C1(F)(CNC(c2cc(CO)no2)=O)CN(C(=O)C=CCO)C1 Cn1ccnc1C(=O)N(CCO)CC.C(C)(C)(CNC(=O)CNC(=O)OC(C)(C)C)N c1(N(CC)Cc2ccc(F)c(F)c2F)ncnc2c1ncn2C(C)C(O)C(F)F N1(CC(=O)N(c2cccc(C)c2)C)CCCCC(C(=O)Nc2cc(C)n(C)n2)C1 N1(C(c2c(N)nccc2)=O)CCCC(NC(=O)CC(C2CC2)C2CC2)CC1 n1(CC(=O)NC2(CC)CCN(C(c3oc(CO)nc3C)=O)C2)cc([N+](=O)[O-])cn1 C1(NC(C(C)(C)c2ccccc2)=O)CCN(C(C2(CC(F)(F)F)CC2)=O)CC1 N1(C(c2ccc(C(C)=O)cc2)=O)CCc2[nH]nc(CNC(c3cnsn3)=O)c2C1 c1(C(N2CC(C)C(NC(C3(C#N)CCC3)=O)C2)=O)cc2n(c1)CCS(=O)(=O)C2 C1(CC(=O)NCC2CC(NC(c3cnc(C(F)F)s3)=O)CC2O)CCCC1(F)F C(=O)(C1=CC2(CCOC2)C1)N1CCC(CNC(=O)C=C2CCCCC2)CC1 N1(C(CN(C(=O)Cc2csnc2C)CC#C)=O)CC=CC1CF c1(C(N2CC(CCNC(=O)CCOCC(F)(F)F)C2)=O)ccc2cnccc2n1 C(=O)(N=c1ccn(CC2CC2NC(=O)C2=C(C)OCCS2)[nH]1)c1c(CC)noc1 C1(CNC(C2(SC)CC2)=O)(CNC(=O)CCCc2cnn[nH]2)CC12CCC2 n1(CC(=O)N(C)CC2C3CN(C(=O)CCF)CC23)cnc2c1CCCC2 c1(CCN(C(C)CNC(c2ccncc2N(C)C)=O)C)cc(F)cc(F)c1 c1(C(=O)NC(C(C)NC(CC(C)C)=O)C)ccc(Cl)cc1 N1(CC(=O)NC2(CCNC(Cc3cn(CC)nn3)=O)CCC2)CCC(C)(O)C1 C1(=O)C(CCF)N1.C(=O)(CCOCC(C)(C)C)N(CC(C)SC)C CC1OC2(CO)CC1(C(=O)NCC1CCCN(C(c3ncc(F)cc3F)=O)C1)C2 C=C1CC2(C1)CN(C(=O)C(C)CNC(C1CCCCCN1C)=O)C2 N1(C(C=C(CC)C)=O)CC2CCN(C(C3C4CCCCCCC34)=O)C2C1 c1(CCNC(=O)CC2(O)CCC2)ccc(-c2nn[nH]n2)cc1Cl c1(NC(C(=O)NC(COC)C2(C)CC2)=O)cc(C)no1 CCC(CC(F)F)C(=O)N(C)CCC1CCN(C(=O)CC2CC2C)CC1 CC1CNCCC1Nc1ccccc1CNS(C)(=O)=O c1(C(C)N(C)C(C2CCCCN2C(c2cncc(F)c2)=O)=O)cccc(Br)c1 C(CCCCCNC(C1(C)CCNC1=O)=O)NC(C=CC)=O C1(C)(OC)CCCN(C(c2ccnc(CNC(=O)C(C)(O)C3CCC3)c2)=O)CC1 C1(N(C(c2scnc2C)=O)CC)CCCN(C(=O)CN2CCS(=O)CC2)C1 N1(C(CCCOC(C)=O)=O)CCCCC1C1CCCN(C(c2csnc2C)=O)C1 C1(C2(O)CCCNC2)(CNCc2c(F)cc(OC(F)(F)F)c(Br)c2)CCC1 c1(C(=O)NC(C(=O)NC(c2cccnc2)CC)C2(O)CCC2)cc(C)c(O)nn1 C12(NC(C3C(C=C)C3)=O)CC3CC(C1)CC(NC(c1coc(C)n1)=O)(C3)C2 C1(C(=O)NCC2CC(F)C2)CN(C(C2CCO2)=O)CC1CN(C)C c1(C(N(C2CN(C(Cc3ccc(NC(C)=O)cc3)=O)C2)C)=O)cccc(Cl)c1O CCCC(C)(O)C(=O)NCC1CCC(CN(C)C(c2ncc(N)nn2)=O)CC1 N1(C(c2c(C)nns2)=O)CC2C(N(C(=O)CNc3ncccn3)C)C2C1 C1(C(=O)NCCC2(NC(=O)CC3CC(F)(F)C3)CC2)CC2COCC(C1)C2(F)F C12(NC(c3ccc(C(=O)OC)[nH]3)=O)CC(C1)N(C(=O)C=C1CCSCC1)C2 N1(C(CC(=O)NCC)=O)CCN(C(=O)CN(C)S(N)(=O)=O)C(CC)C1 C(=O)(C1CCOc2ccccc21)NC(CNC(c1ccc(C(C)C)o1)=O)(C)C Cc1nc(C2CC2)sc1CC(=O)NC1(C)CC(NC(C2CC(C)(C)C2)=O)C1 C12(CC(=O)N(C3CCN(C(=O)Cc4cnsc4)C3)CC)CCC(CC1)C2 C1(CNC(=O)COC2CC=CC2)CN(C(=O)C2=NNC(C(F)(F)F)C2)CCCO1 N1(C(c2cc(CC)n(C)n2)=O)CC(C)(C)CC1C(=O)NC1CC=CCC1 c12ocnc1C(=O)NC2.C1(C(=O)NCCN(CCC)CC)CCC(C(N)=O)O1 CC(CC#N)C(=O)N(C1(C(=O)NC2CCCSCC2)CC1)C C12(C(=O)OC)CCC(C(=O)N=c3[nH][nH]cc3NC(COC)=O)(CC1)CC2 c1(C(=O)Nc2nc(C(N3CCC(C(=O)OCC)C3)=O)n(C)c2)ccc(Cl)c(O)c1 N1(C(c2cc(C#N)[nH]c2)=O)CC2CCOCC2(NC(=O)C2=CCCCCC2)C1 c1(C(N2CC(C(C)NC(=O)C(C)(F)F)C2)=O)cncc(F)n1 C1(NC(=O)NC2CCCC(OC(C)(C)C)C2)COc2cscc2O1 c1(COC)cnc(N2CCCC(NC(c3coc(Br)c3)=O)C2)nc1 C1(N(C(Cn2c(C(C)C)nnn2)=O)C)CCN(C(=O)CC2CC3(CC3)C2)CC1 CN1CCC(=CC(N2CCC(CNC(c3ccnc(Cl)c3)=O)C2)=O)CC1 c1(CC(=O)NCC2(NC(C3CCC4CC34)=O)CC2)cccc(Cl)c1F C1(NC(=O)C=CCO)(CNC(C2CCCC(F)C2)=O)CCOCC1 n1(CC(=O)N(CC(=O)N(CCCF)CCO)C2CC2)cncn1 CC1(NC(c2cocn2)=O)CCN(C(C2CC(C(C)(C)C)C2)=O)CC1 C12(OC)CCCC(C(=O)NC3CC4(C3)CN(C(C3(OC(C)=O)CC3)=O)C4)(CC1)C2 C1(C(N2CC(OCCOC)C2)=O)CN(C(=O)CCCC2CC2)CC12CCC2 C1(O)(CCOC)CN(C(=O)CC2CC2CNC(=O)CCOCC(C)C)C1 C1(NC(C(CC)F)=O)CC2(NS(=O)(=O)Cc3cccc(SC)c3)COC1C2 C1(NC(C=C(COC)C)=O)COCCC1NC(=O)C(C)NC(C1CN(C(N)=O)C1)=O C(=O)(CCS(N)(=O)=O)N1C(CCN(C(c2oc(CC)c(C)c2)=O)C)CCCC1 c1(C(=O)NC2CN(C(C(C(C)(C)C)OC)=O)CC2C)nc(Cl)c(=O)[nH]c1N Cc1cc(C(=O)N(C)CCOCCN(C)C(c2ncsc2C2CC2)=O)cc(C)c1 c1(OC)cc(C(N2CC(NC(c3c[nH]c(C)c3)=O)CC2(C)C)=O)ccc1C c1(CNC(C(c2scc(CCC)n2)N2CC3CC2C3)=O)ccccc1Cl N1(C(C2CC(CC)(CC)C2)=O)CCCC1(C)CNC(=O)C(C)Oc1ccccn1 Cc1cnc(S(C)(=O)=O)nc1N1CC(C(=O)NCC(C)(C)F)CC(F)C1 Cc1[nH]nc2c(C(=O)NC3CCC(CNC(C4(C#N)CCOC4)=O)C3)cccc12 Cc1sc(C(C)C)nc1SC(CCNC(c1ccc(C(=O)N(C)C)cc1)=O)(C)C C#Cc1ccc(C(=O)NC2(C(=O)NC3CCOCC3F)CCC2)nc1 O=C(N=c1[nH]n(C(F)(F)F)cc1Cl)NC(c1cccnc1-n1cncn1)=O N1(C(CC2(C)CC2(F)Cl)=O)C2CCC1CN(C(=O)COC1CCCC1)C2 c1(C(N2CCC(N(C(=O)CC3CCCCC3)C)C2)=O)ccc2c(c1)C(=O)CCC2 c1(CC(=O)NCc2c(C(N(C(CC)COC)C)=O)cco2)cccc(F)c1 C1(C(N2CCC(NC(CC(=O)NCC(F)(F)F)=O)C2)=O)CCC2(CCOCC2)O1 c1(NC)ccc(N=c2ccn(CC(=O)OC)[nH]2)cc1C(F)(F)F c1(C2(C(N(CCNC(C(C)SCC)=O)C3CC3)=O)CC2)oncc1C C(=O)(C(C(C)(C)C)SC)NC1C(CNC(c2nc(CCC)oc2)=O)COC1 C#CCC(CC#C)C(=O)N1CC(CNC(=O)CC(C)F)(OC)C1 c1(C(=O)NC2CC2NC(C2CC2[N+](=O)[O-])=O)[nH]c2ccccc2c1Br N1(C(c2c(CC)occ2)=O)CCC(C)C(CNC(=O)C(C)NC=O)C1 C1(C(N(CC=C)C)=O)COC2(CCN(S(=O)(=O)c3cccnc3Cl)CC2)C1 C1(C(=O)NC(c2cc[nH]n2)C)(NC(=O)OC(C)(C)C)CC(F)C1 c1(CCC(=O)N(CCCCN(C(C(CC)SC)=O)C)C)ccc2ccccc2n1 C(=O)(CCCOC)NC(C)C(C)C.C1CC(=O)N1CC C(c1ccncc1C)=CC(=O)N(C(CN(C(C1N(C(=O)OC)CCC1)=O)C)C)C c1(-c2n(C3CCC(C)C3)nc(CC3CC3)n2)ncnc2c1c(Br)cn2C N1(CC2(CNC(C3(O)CCCCC3)=O)CC2)CCC(NC(C2C=CCC2)=O)CC1 C1(CNC(CCNC(c2ccncc2)=O)=O)CN(C(C2(Cl)CC2)=O)CCC1(F)F CC1CCCN(C(=O)CC2CC2)C1CO.C12CCCN1C(=O)C21CC1.c12cc-1on2 C12(CC)CN(C(=O)OC(C)(C)C)CC(F)(C1)C2.c12ccc(cc1)C(C)(O)CN2 c1(NCCC(C)F)nccc(N(CC(F)(F)Br)C)n1 Cc1cccc2cc(C(N3CCC(C)(NC(c4csnc4Cl)=O)CC3)=O)oc12 C(CC(C)C(=O)N(CCC(C(C)C)NC(c1csc(CO)n1)=O)C)=CCC C(=O)(NN=c1ccc2nccn2[nH]1)c1c2ccn(CCN(C)C)c2ccc1 CN1CCN(C=O)CC1C1CC1.c1(C(CCN)=O)nc[nH]n1 N1(C(C=CC(C)NC(=O)C(C)(O)C2CCC2)=O)CC(=O)NC2(CC2)C1 C12(CNC(c3nc(N(C)C)oc3)=O)CC(CCO1)N(C(=O)CCn1cccn1)C2 CCCCCCn1nnnc1C(C1CCC(=O)O1)NCCCOCC1CCC1 c1(CC(=O)NCC2CN(C(C3CC(SC)C3)=O)CC23CC3)cnc2ncccn12 CS(=O)c1ccc(-c2cn(CCCCCNC(=O)C(C)(Cl)Cl)nn2)cc1 C1(CNC(C=C(C)C(C)C)=O)CCCC(CNC(C2CCC(=O)CC2)=O)C1 c1(C(=O)NC(C)CNC(c2ccco2)=O)cnc2ccnn2c1N c1(C(=O)NCC(C)(C)NC(CC(C)NC(N)=O)=O)cc(F)ccc1O.C(CO)O c1(C(C)N(C(C)C(=O)OCC2CC2)C2CC2)ncc(Br)s1 C12CN(CC1CC)C2=O.n1(CCC)cc(CNC(c2noc(C)n2)=O)cn1 C(=O)(CCN=C(NC(c1ccc(C)o1)C)NC(CC)CC)OCC#C CC1CC(C)N(C(c2cc(S(N)(=O)=O)c[nH]2)=O)CCN1C(c1cc[nH]c1)=O CC1CCCN(C(C2CCCN2C)=O)C1CNC(C1(F)CC1c1ccccc1)=O C1(C(=O)NC2(C(F)F)CC(NC(C3CN(C)C(=O)N3)=O)C2)CC2(C1)CC1(CC1)C2 Cn1[nH]c(C(=O)NC2CCCCC2NC(C2CC2(C)C(F)(F)F)=O)nc1=O CN(OCC(F)(F)F)C(=O)C(F)CC1CC1.C1(C(F)(F)F)(C(=O)N)CC1 c1(C(N(C)CC2CCCN(C(c3c(CC)[nH]nc3Cl)=O)C2)=O)cc2scnc2[nH]1 N1(C(C2(C(=O)OC)CC2)=O)CC(NC(c2ccnc(N(C)C)c2)=O)C2(COC2)C1 c1(C(=O)NC(C)CC(C)NC(C2CC3CC2C2CC32)=O)ccc2c(c1)nnn2C c1(CCNC(=O)COCC2CC2)c[nH]nc1O.C1(N)CCCC1 c1(C(N2C(C)CN(C(=O)CSC(F)(F)F)CC2)=O)ccc2[nH]nc(O)c2c1 C1(NC(=O)C2=COCCC2)CC12CCN(C(c1cc(F)ccc1N)=O)CC2 C(=O)(C(C)(C)CSC1CC1)NCCNC(CCN(CCCCC)CCC)=O O=Cc1sc(CNC2CN(C(c3cc(Cl)cc(Cl)c3)=O)CC2C#N)c(Br)c1Br C(CCCCCC(=O)N1CCN(C(c2ncc(F)cc2F)=O)CC1)SC C=CC(F)(F)C(=O)NCCCCCCNC(=O)C=CC Cn1[nH]c(C(=O)NC(C)(CNC(=O)Cc2cc[nH]c2)C2CC2)nc1=O CC(C)CC(C)C(C(=O)NCC1CCCO1)N1CC(=O)NC(C(C)C)C1 c12ccc(cc1C)o2.N1(CC(=O)NCC)CCSCC1C1CCC1 C1(NC(CCN(C)CC)=O)CC(C)CN(C(=O)CCCCCSC)C1 N1(C(C(CSC)C)=O)CC(C(=O)NCCCn2ccnn2)C(C)C1 C1(NC(C2CC2F)=O)CC2CCC(C1)N2C(c1cc2cc(Br)sc2[nH]1)=O C1(NC(C(C)NC(N)=O)=O)CC2CC(C1)N(C(=O)COc1ccccc1)C2 c1(CNC(C2(C#N)C(C)C2)=O)ccc2c(c1)CCN(C(=O)C(C)(Cl)Cl)CC2 c1(C(N2CCC3CCCC3C2)=O)cc2nc(Br)sc2[nH]1 C1(C(=O)NCC(c2ccccc2F)NC(c2c(C)ncs2)=O)C2CNC(=O)C12 N1(C(C(C(C)C)N(C)C)=O)C2CCC1CN(C(=O)C(=Cc1cn(C)nn1)F)CC2 c1(C(=O)OC)ccc(C)c(CO)c1.c12ccc(cc1)C(C)NC(=O)C(=O)NC2C CC(C)C(CC(=O)N1CC2(CC(NC(C3OCCN(C)C3=O)=O)C2)C1)C(C)C C#CCC(CC(=O)NOCCF)NC(=O)C(C)CC(C)CC S(=O)(=O)(c1ccc(NCC(C)Cn2cccn2)c(Cl)c1)NC(CC)CO c1(C(=O)NCC(CN(C)C(c2csc(C(N)=O)n2)=O)(C)C)cc2[nH]ccc2s1 c1(C(=O)NC(CN(C(C2C(COC)(COC)C2)=O)C)(C)C)cc([N+](=O)[O-])oc1C C1(O)(CNC(C(CC)CC)=O)CCCN(C(C2(C#N)CC3CC3C2)=O)CC1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)NC(C1CC(Nc2nc(Cl)nc3ccccc23)C1)=O C=CC1CCCCN1C(C12CC1CCN2C(=O)C1=CCCCC1)=O Cc1ccccc1C1C(O)CCN1C(C1CN(C)C(=O)N1)=O C1(CNC(c2c(C)nc(-c3ncc[nH]3)s2)=O)CN(C(C2CC2(F)F)=O)CC12CC2 Cn1cc(C(C(=O)NCCCOCC(F)F)NC(c2ccc(Cl)o2)=O)nn1 c1(C2C(=O)N2)cnn(CC2CC2)c1.C1(N)CCCC1.C(C(C)C1CC1)N(CC)CC C1(C2CCC2)(C(=O)OC)N(C(=O)NC(c2n[nH]c(C)n2)COC)C1 N12CCC(CC)(CC1)C2=O.c1(CNC(C2CC(=C)C2)=O)ccc(NC(C)=O)nn1 C(=O)(C#CC1CCCO1)N1CC(c2ccccc2)(NC(c2coc(Br)n2)=O)C1 C(=O)(C1=COCCO1)N1CC(SC)C(NC(=O)C(C)(O)Cc2ccccc2)C1 c1(CC)cc(C)c(C(=O)N(CC(=O)Nc2cn(C)nc2CC)CC)o1 C(=O)(C#CC1CCCO1)N1CC(O)(CCNC(C2CCCCC23CC3)=O)C1 C1(F)(Cc2cn(CC3C(N(C)C)CN(Cc4nncs4)C3)nn2)C(C)(C)C1(C)C C1(COC)CN(S(C)(=O)=O)C1.C12(CC1)CC(=O)N(C1CC1)CCCNC2=O C(=O)(C(CC(C)C)ONC(c1ccncc1F)=O)N(C)Cc1occ(C)c1 C1(NC(CSCC)=O)COC2(CCN(C(=O)C(C)SC)CC2)C1 C(CCC(=O)NC1CCC(CNC(=O)COC(C)C)C1)OCCOCC c1(C2C(C(=O)NCC(C3CC3)NC(C3C=CCCC3)=O)C2)ccc(F)cc1 N1(C(C(C)CC2CCCC2)=O)CCc2c(CNC(=O)CSC3CC3)cccc2C1 Cc1cc(C(N2CCC(C)(NC(C3CC(F)C(=O)N3)=O)CC2)=O)cc(F)c1C c1(NC(C2N(C(c3ccc(C)c(Cl)c3)=O)CCOC2)=O)c(Cl)ncc(Br)c1C c1(C(N(C)CC2(NC(C(CSC)O)=O)CC2)=O)cccc2c1NC(=O)CO2 C(=O)(CN=S(C)(C)=O)NC(CN(C(=O)C#CC1CC1)C)Cc1ccccc1 c1(NC(=O)C2=CCCN(Cc3ccc(Cl)s3)C2)cccc2c1OCCC2 C1(OC)CC(C(N(C)CC2CCN(C(c3cnc(OC)nc3)=O)C2)=O)N(CC)C1 c1(OCC(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)cccc(C#N)c1 Cc1cnn(C)c1CNC(=O)CN(C)C(c1csc(F)c1)=O N1(C(c2c(C)nccc2)=O)C2CCC1CC(O)(CNC(=O)C1=CSCCO1)C2 N1(C(c2cc(C)c(F)cn2)=O)CCCN(C(=O)CCc2cnc(O)[nH]2)C(C)C1 C1(CCCC)CN(N(Cc2ccc(OC)nc2)Cc2ccc(C(=O)O)nc2C)C1 N1(C(c2n(CC)nc(C)c2)=O)CCCCC(OC)C1 n1(CC(=O)NCC2C(NC(CC3(OC)CCC3)=O)C2)cc([N+](=O)[O-])nc1C c1cccn1C.n1(C(=O)NC(C)CNC(=O)CON2CC=CC2)nnnc1C1CC1 c1(C(=O)NCC2OCCCN(c3c(CC)cccn3)C2)c[nH]c2c(F)cccc12 Cc1c(CN2CCOC(CNC(C3(CC(C)C)CCC3)=O)C2)cnn1C N1(C(Cc2c(C)noc2Cl)=O)CC2CS(=O)(=O)CC2(NC(=O)C=CC(C)(C)C)C1 C(C)(CCCCNC(c1ccccc1)=O)NC(c1cc(C(CC)C)no1)=O N1(C(=O)NCC2(C(F)F)CCOCC2)CCC(Cc2ccc(I)cc2)CC1 C(CCCCNC(=O)CSS(C)(=O)=O)N(C(=O)CSC(F)F)C N1(C(c2cn(C(C)(C)C)nn2)C(=O)NC(C)C)CC(CO)OC2(CCC2)C1 N1(C(CNS(N(C)C)(=O)=O)=O)CC(OC)CC(CO)C1.c1(CC(=O)N)c[nH]nc1O CC1COCC1N=c1nc2sccc2c(N)[nH]1.C(C(C)(C)C)NCC CCS(=O)CC(=O)N1CC(NC(=O)C(=O)Cc2ccccc2)CC1C N1(C(C2C(C)C2)=O)CCCC2(NC(c3coc(-c4ccccc4)n3)=O)CC2C1 N1(C(C2OCCN(C(C)C)C2)=O)CCN(C(=O)C(C)CCO)CC(O)C1 N1(CC(=O)NC2C(NC(CCc3nc(C)sc3)=O)CCC2)CCc2ccccc21 c1(C=O)ccc2c(c1)C(C)C(C)O2.C1(OC)(CNC(=O)CC)CCN(C(C)=O)CC1 N1(C(CSc2n[nH]c(O)n2)=O)CCC(C(=O)O)CC1.n12cc(nn1)CNC(=O)C2 Cc1cccc(N2CCC(NC(=O)NC3(CN(C)C)CC3)C2=O)c1 N1(NC(c2cn(C)nn2)=O)CCC(CCC2CCCN2C(=O)Cn2cnnc2)CC1 CCCC(CC(C)C)C(=O)NC1CCC(CC(=O)NC2CCC3(CC3)C2)C1 N1(C(C(COC)NC(C)=O)=O)CCN(C(C2(CC(C)C)CCC2)=O)C(C)C1 C1(CC)CCCC1(C)C(=O)N(CC(=O)NCC(C)(C)n1ccnc1)CC1CC1 c1(NC(C2CC(NC(CNC(=O)NC)=O)C2)=O)ccc(-c2ncn(C)n2)cc1 c1(NCC)ccc(CNCC(O)Cc2cccc(F)c2)cc1 CSC1=C(C(=O)NCC2CCCN2C(=O)COCCF)CCCC1 c1(C(=O)NC2CN(C(C3CCCC3C(F)F)=O)C2)cc2c(Cl)ccc(Cl)c2[nH]1 c1(OCCOC(c2ccc(-c3cc[nH]n3)cc2)=O)ccc(F)c(F)c1 C(CCC(=O)NO)NCC1C(N)CC1 Cn1cnc2cc(C(=O)NCC3(O)CC(CNC(=O)Cc4nc[nH]n4)C3)ccc12 Cc1c(C(=O)NCC(C2CC2)NC(=O)CCCCC2CC2)cccc1S(N)(=O)=O C1(CCC(=O)NC2CCCC(SC)C2)CCc2ccccc2C1=O CCC(CC)(CO)C(=O)NCCC1CC(NC(C2CCC(=O)N2C2CC2)=O)C1 CCC(CCC(=O)NC1CCCC1C#N)NC(C1(C)CSC1)=O c1(C(c2nnnn2C)NCCSC)cc(C(F)F)ccc1N1CCCCC1 c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)ccc2c(c1)CCC(=O)N2 N1(C(c2c(CC)nccn2)=O)CC(NC(C2OCCO2)=O)CC12CCCOC2 c1(NC(C2CCN(CC3CC3)CC2)=O)ccc(Br)cc1O c1(C(=O)NC2CC(C(=O)NC(c3nc(=O)o[nH]3)C)OCC2)ccccc1N(C)C C(=O)(C(CC1CC1)NC(=O)CONC(=O)Cn1ccnc1)OC N1(C(C2CN(C(C(C)SC(C)C)=O)CC2C)=O)CC(C(N)=O)CC(C)C1 C1(COC)(CC2CC2)CC=CC1.C1(=O)CN(C(C2CSC2)=O)N1 C1(CC(=O)N(C(CC)C)CC)CN(C(=O)CSCC(F)F)CCO1 C12(SCC)CN(C(=O)OC(C)(C)C)C(CNC(=O)CC3(C)CCS(=O)(=O)N3)(C1)C2 c1(C(=O)NC2CCC(CNC(CN(C3CCC3)C)=O)CC2)cc(=N)[nH]c(Cl)n1 c1(CC(=O)N(CCNC(C(c2cccc(Cl)c2)C)=O)C2CC2)ccccc1Cl CC1CC(OC(c2cnccc2C(F)(F)F)=O)CC(C)(C)C1 Cc1nc(C(=O)C(=O)NC(C)(CNC(=O)CN(C)C)Cn2cccn2)cs1 c1(C(C(=O)NC(C)C)N(C2CCC(C)(C)C2)C)ccc([N+](=O)[O-])cc1 C(C(Cl)C(=O)N1CCC(CC(N2CC3CC3C2)=O)C1)OC C1(NC(Cn2c(C)ncc2)=O)CCN(C(=O)Nc2cccc(Cl)c2Cl)C(C)C1 C1(NC(C(=O)N(CC(c2ccccc2)O)C)=O)CC2CCC(C1)N2CC1CC1 Cc1ccc(C(N2CCC(NC(C3CC3c3cccnc3)=O)C(F)C2)=O)cc1Cl C1(C(N2CCC(N(CCC)C(c3cnn(CC)c3)=O)CC2)=O)CCCC(=O)O1 N1(C(C=C(C)C(F)F)=O)C2CC1CN(C(C1(CO)CCCC1)=O)C2 CC(C)C(CCN(C)C(C1CCCC1(F)F)=O)NC(=O)COCCCN(C)C CC1(C)COCCN1C1CC(C(=O)NC2(c3ccc(C(F)(F)F)c(F)c3)CC2)C1 c1(C(N(C2CCCC(NC(c3cncc(OC)c3)=O)C2)C)=O)cc(N)c(F)cn1 C(=O)(CCC(F)(F)C(F)(F)F)N1C(C(C)NC(C2CCC(C)(C)CC2)=O)CCC1 C1(CNC(C2(OC)CCSC2)=O)(CO)CCCN(C(=O)COc2ccn(C)n2)C1 C=CC1(C(=O)NC(C)CC2CCN(C(c3cn(C)cn3)=O)CC2)CCOCC1 Cc1c[nH]c(C(=O)NCC(CC(C)C)NC(=O)COc2cccnc2Cl)c1C c1(OC)cnc(C(=O)NC(C(C)NC(c2n[nH]c(C)n2)=O)C(C)C)nc1 Cc1cc(CC(=O)NCCCC2CCCN2C(=O)C(=O)NC2CC2)ccc1CO Cc1ccc(CC(=O)N(C)CC2CCN(C(=O)C(C)OC(C)(C)C)C2)c(F)c1 CC(C)C(CC(=O)N1CCOCC1CN(C)C(c1cncn1C1CC1)=O)C(C)C C1(C(=O)NC2(C3CN(C(C4=NOC(C)C4)=O)C3)CC2)CCc2ncccc2C1 C1(CC=C)(C(=O)NCC2CC2NC(=O)C(O)Cc2ccccc2)CCCC1 N1(CC)CCCN(C(=O)C(C)(C)C(C)NC(=O)CCCCCOCC)CC1=O Cc1ncc(C(=O)OCc2cc(Cl)ncc2Cl)c(Cl)c1Br C=CCC(CC=C)C(=O)NCC1CCN(C(C2CNC(=O)C(C)(C)C2)=O)C1 c1(CNC(C2CN(C(=O)OC(C)(C)C)CC(C)O2)=O)cncc2ccc(F)cc12 C1(C(N2CC(CC(C)NC(=O)C=CC(C)(C)C)C2)=O)CCCCCCC1 N=c1[nH]c(C(N2CCC(CCNC(=O)COC3CCCOC3)C2)=O)cs1 C1(NC(c2ccc(C)s2)=O)CN(C(=O)Cc2ccc(Cl)cc2Cl)CC2CCCC12 C(=O)C(C(C)(C)O)c1ccccc1.CC1(C)CCNC1 C=CC(C)(O)CC(=O)NCc1ncccc1C(=O)NOCCc1ccccc1 C=C(Cl)CC(C(=O)NCc1nccc(OCC)n1)NC(=O)C(C)OC1CCCC1 CC(CCCCNC(=O)C(C1CCC1)C1CCC1)NC(=O)CC1CC(=O)NC1=O S(=O)(=O)(c1c[nH]ccc1=NCCC(=O)Nc1ccccc1)CC(=O)NC C1(N(C)C)CC2(CCN(C(=O)CCN3CCN(C(=O)CCBr)CC3)CC2)C1.C(CO)N C(C(C(C)(C)C)NC(=O)CCCN1CCC1)NC(CCCN(C)C)=O CC(=O)CCCC(=O)NCCC(O)C(=O)N1CCCOCC1 C(=O)(C(C)S(=O)(=O)C(C)C)NCCC(C)N(C(C(CC(=C)C)NC(C)=O)=O)C Cc1cccc(CCSC(C)C(=O)NC2CC(NC(=O)C(C)OC3COC3)C2)c1 C=CC1CN(C(=O)CCNC(=O)C(C2CCCC2)OCC)CCO1 N1(C(C2(CCC)CCNC2=O)=O)C2CCC1CC(NC(c1cc[nH]c1)=O)C2 N1(C(c2c(C)cc(C)nc2O)=O)CC2(CCC(NC(=O)CCCC(C)O)CC2)C1 N1(C(C(CC)C(C)C)=O)CC2(CNC(c3ccco3)=O)CCC1CC2 CCC(Cc1ccccc1)CC(=O)NCCCN(C(=O)CC(O)CN(C)C)CC C1(CCCC)CCCC1(c1nnnn1C1CC1)NCC(C)(C)CCO C(=O)(CS(=O)(=O)N1CCCCC1)NC1CCN(C(CCCOCCC)=O)C1 CC(C)C=CC(=O)N(CC(N1CCC1)=O)CCO.C(C)C CN1N=C(C(=O)NCCCCC(O)C(=O)N2CCCNC(=O)C2)CCC1=O C1(NC(=O)C(O)C2CN(C(=O)CC3CC=CCC3)C2)COC2(CCCC2)C1 CC1CCC(C)(C(=O)NC(c2ccccc2F)CNC(=O)Cc2cn(C)nn2)C1 N1(C(C(=Cc2cnc[nH]2)C)=O)CCC(NC(=O)COCc2nccs2)C(O)C1 c1(C(N2CC3(CC(NC(c4cnc(SC)nc4)=O)C3)C2)=O)cc(C)c(Cl)c(C)c1 c1(C(N2CCCC(NC(=O)CC3CSCCS3)C2)=O)cc(F)cc([N+](=O)[O-])c1 CN1CCc2[nH]nc(C(N3CCC4C(NC(=O)CCCC#N)C34)=O)c2C1 CC1=NC(C(=O)NC(C)CN(C)C(c2ncn(-c3ccccc3)n2)=O)CS1 C(=O)(C(C(C)C)(C(C)C)N(C)C)NCC1CC(OC)CN1C(=O)C=C(C)C(C)C C1(NC(c2c(C)noc2C)=O)C2CCCN(C(C34CC(F)(C3)C4)=O)C2C1(C)C C=CCC(C)(O)C(=O)N1CCC(C(C)C(N2CCOC(C(C)(C)C)C2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)N(C1CC(C(N(C(C)C(N)=O)C)=O)C1)C C(=O)(CCCC(C)(C)NC(C1CC(=O)C12CCC2)=O)N(C1CCCCC1)C S(=O)(=O)(c1ccccc1)C(CSCC(=O)NC(C1CC1)CNC(CC(C)F)=O)=O c1(CC)ncc(C(c2nnnn2C2CCOC2)NCC(C)(C)OC(C)=O)[nH]1 CS(=O)(=O)c1cccc(CNC2(c3nnnn3CCCF)CCCNC2=O)c1 C(=O)(C#CC1CCCCC1)N(C)CC1CCCCN1C(=O)C(=O)NCCC(N)=O C1(NC(C2(CCCC)CCC2)=O)CN(C(C2(CF)CC2)=O)CC1O C(C(=O)NCC12CC(CNC(=O)CCC(C)SC)(CO1)C2)(C(C)C)OCC c1(C(=O)NC(C2(O)CN(C(=O)CC3CCOCC3(C)C)C2)C)ccn2cccc2c1 N1(C(C2N(C)CC2)=O)CC(C2CCN(C(=O)C3=NOC4(CCOC4)C3)CC2)C1 C1(CCCC)CCCN(C(c2cc(OC)ns2)C(=O)NC2CC2)C1.C(COC)S c1(N(C(=O)NCCN2CC=C(C)CC2)C)cccc2nsnc12 C(CN=C(NCc1cnco1)NC1CCN(C(=O)N(C)C)CC1)OCC C1(CNC(Cc2scc(C)c2)=O)CN(C(c2csc(C)c2N)=O)CCC1(C)C c1(CC)cccc(C(=O)NCC2CCN(C(=O)CCSCC(C)C)CC2C)c1C Cc1nn(C)c(N)c1C(=O)NCC(C)(C1CC1)NC(=O)CN1CCOCC1=O c1(C(=O)NCC2C(CNC(c3ccc(CC)[nH]3)=O)C2)nc(=O)n(C)[nH]1 N1(C(c2c(C)oc(CNC(=O)Cn3cnnc3)n2)=O)CCC(C)(O)CC1 C#Cc1cnn(CC(=O)NCC2C3CN(C(C4CC4C(N)=O)=O)CC23)c1 N1(C(C2CC(C#N)C2)=O)CCN(C(C2CC3C=CC2O3)=O)C(C2CCCC2)C1 c1(C(=O)NCC2C(NC(CSCCC#N)=O)C2)coc2c1C(=O)NCCC2 N1(C(c2cn(CCC)nc2)=O)CC(NC(=O)C(N2CCOC2=O)C)C(C2CC2)C1 C1(O)(CNC(COC)=O)CCN(C(c2ccoc2Cl)=O)C1 N1(C(C2(CC)CC2(F)F)=O)CCC2CN(C(=O)CCC3CCC(=O)N3)CC2CC1 C1(NC(C(N2CCC(CC(C)C(=O)O)CC2)=O)=O)CCc2ccccc2C1 C(c1ccccc1F)=CC(=O)NC12CN(C(c3cn(CC=C)nn3)=O)C(C1)C2 Cc1cc(C(=O)N(C(C)CCNC(=O)CCCc2csc(=N)[nH]2)C)sc1C c1(C(N2CC(CC(C)NC(C(CC)CC)=O)C2)=O)ccc2cnccc2n1 O(NC(=O)C(Cc1cc[nH]n1)NC(=O)Cn1cnc(C#N)n1)CC1(C)CCCC1 C=CC(C)(C)CCNC(C1(C)CCN(C(C2(O)CCSCC2)=O)C1)=O N1(Cc2cn(C)nc2)CCN(C(=O)C(=O)NC(CC(N)=O)C2CCOCC2)CC1 c1(CC)cc(F)c(C(=O)NCC2COCC2NC(=O)C=CCOC)cc1F C1(C#N)(OC)CC(C(N2C(C(=O)NOCC3CC(=O)NC3=O)CC2C)=O)C1 c1(C(=O)NC2(CCNC(=O)CSCC(F)(F)F)CC2)nnc(O)nc1O c1(OC)cc(C2CC2)ccc1C(N1CC(Cc2cn(CCC(F)(F)Cl)nn2)C1)=O N1(C(c2cnc(CC)[nH]2)C(=O)NCCCC2CC2)CCC(C(C)(C)C)CC1 N12CCCCC1c1ccc(cc1)C(=O)NCC2.c1(N)ccccn1.C(=O)O N(C(=NCc1ccccc1Cl)NC1CCC1)CC(C1CCCC1)OC c1(CN2CC(O)(CNC(=O)CC3CCOCC3)C2)c[nH]c2cccnc12 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCC(NC(=O)CC2CCCO2)C(F)C1 N1(C(Cn2c(C)ccn2)=O)CC2(CCCCN2C(c2cc(F)cnc2O)=O)C1 CC(C)CCC(O)C(=O)NC1(CNC(C2CCc3nncn3C2)=O)CCCCC1 Cc1c(C(=O)NCC2CC3CN(C(c4ccsc4)=O)CC23)sc2nnc(S)n12 C(CC1CC1)(C(=O)N(C)Cc1ccncc1)NC(CNC(CCC)=O)=O c1(CN(C(=O)CC2(NC(=O)OC(C)(C)C)CCOC2)C)c(C(=O)NC)cnn1C CCCCCCC(CC)C(=O)NCC1COCCN(c2cc(C)c(C#N)cn2)C1 C12(CCNC(C(C)NC=O)=O)CCC(C1)N(C(c1ccc(Cl)nc1O)=O)C2 C1(C(=O)NCC(C)CN(C)C(C2(C)CC(C)(C)C2)=O)CCC(C)(C)CO1 c1(C(=O)NCC2(C)CCN(C(=O)Cn3cccn3)C2)ccnc2c(F)cccc12 c1(OC)ccc(Cn2nc(Br)nc2Cc2cccc(OC(F)F)c2)cc1C(C)C CCCCCCC(C)C(=O)NC(C1CCCN1C(c1ccc(=NCC)[nH]c1)=O)C C1(C(c2cn3c(n2)CCC3)C)CCCCN(C(=O)C(C)(C)c2ncco2)C1 N1(CCCNC(C2(CCC)CC2)=O)CCN(C(=O)CC(C)CC)CC1 C(=O)(C1=CC(C)CC1)N(CCNC(=O)Cc1ccc(-n2nccc2C)cc1)CC c1(C(=O)NC2(C)CN(C(=O)CCCc3nccs3)C2)cc[nH]c(=N)c1 c1(CNC(c2csc(CC)n2)=O)cc(C(=O)NCc2scc(CCC)n2)n(C)n1.CC C1(N(C2CCN(CCNC(C(CN(C)C)O)=O)CC2)C)CC12CCC(F)(F)CC2 c1(C(N2CCCC(NC(c3nn(CC)c(C)c3)=O)CC2)=O)cccc2oncc12 C1(C(=O)NCCOC2CN(C(C(=O)N(C)C)=O)C2)CCN(S(C)(=O)=O)CC1 N1(CCCN(c2ccc(Cl)cc2)C(c2ocnc2C2CC2)=O)CCCCCC1 CC1CC(NC(C2COC2)=O)CCN1C(=O)COc1ccc(F)c(Cl)c1 c1(Cn2cc(C(N(C(Cc3ncc(C)nc3)=O)C)C)nn2)ccc(Cl)cc1Cl C1(C#N)(C(N(CC(CNC(CC(C)CN(C)C)=O)(C)C)C)=O)CCCOC1 C1(NS(C)(=O)=O)CC2(CCC(CN3CCC3C(=O)NC(=O)CNC(N)=O)OC2)C1 C1(CNC(C(C)C)=O)CC(C(F)(F)F)CCN1C(c1cc[n+]([O-])cc1)=O c1(C(=O)NCC(C2CCOC2)NC(c2n(CC)ccc2)=O)nn(C)cc1[N+](=O)[O-] c1(OC)cc(NC(=O)Cc2ccc(-n3cc(-c4ncoc4C)nn3)cc2)ccn1 C(=O)(CC(O)C(C)(C)C)NC1CCN(C(C2(NS(C)(=O)=O)CC2)=O)CC1 C(=O)(C(F)(F)CNC(C1CN(C(c2cc(C3CCC3)no2)=O)CC1C)=O)OC C(=O)(C1CSc2ccccc21)N(C1CN(C(CCCC#CC)=O)CC12CC2)C N1(C(C)C)CCCC(C(N2CCCCC2)=O)C1.c12ccc(cc1)NC2 c1(OC)cc(F)ccc1C(N1CCCC(C)C1CNC(=O)Cc1ccsc1Cl)=O C1(CC#C)CN(C(C2CCC(C(C)C)N2C(c2ncccc2C)=O)=O)CCO1 c1(SCCC(=O)NCCNC(Cc2c(C)occ2)=O)cc(F)ccc1F C1(CCOCC)(C(=O)N(C)CCN(C)C(C2(CC)CCC2)=O)CCCC1 CC(C)(F)CCC(=O)NCC1CC1CNC(c1cc2occc2[nH]1)=O c1(C(C)(F)F)cccc(C(N2CCOC(CNC(c3cscc3C#N)=O)C2)=O)c1 Cc1cc(C)cc(NNC(=O)C(=O)N2CCCCC2)c1 c1(NCC(C2(OC)CCCCCC2)=O)cc(OC(F)F)c(Br)cc1C Cc1ccc(-c2ccc(C(N3CCCC3c3ccncc3C)=O)o2)cc1 C(CCC(C(=O)NCc1cc(C)no1)NC(=O)CC1CCCCCC1)OC N1(C(CSCCCC)=O)CCN(C(=O)C=CCCc2ccccc2)CC1C(C)C c1(-n2cc(C(CC(=O)Nc3c(C)nccn3)O)nn2)cc(F)c(F)cc1F N1(C(C(=O)NC2CCCCC2)CC2CCC2)CC2CC(C1)c1cccc(=O)n1C2 N1(C(C2C(OC(C)(C)C)C2)=O)CCCC(C2CN(C(=O)C(F)(F)c3nccs3)C2)C1 C1(CNC(C(C)(C)n2cnnn2)=O)CC2(CO1)CN(C(C1CCC1(F)F)=O)C2 c1(N(C)CCOC2CC2)nc(N2CC3OCCOC3C2)nc2scnc12 C1(C(=O)NCCc2onc(C)n2)CC2(CC(NC(c3cc4n(n3)CCO4)=O)C2)C1 c1(C(N2CC(NC(CC(CC)SC)=O)C(C)(C)CC2)=O)cccc2[nH]cc(Cl)c12 c1(OC)cc(C)ccc1C(=O)NC1CS(=O)(=O)CC1NC(c1n[nH]c(C)c1O)=O C=CCCCC(C(=O)NCC1CC(=O)N(C)C1)NC(=O)CCOC(C)C N1(C(CCCOC)=O)CCN(C(c2ccnn2COC)=O)C2CCCCC2C1 C(CCC(O)C(=O)NCC1CCCCO1)NC(C1(OC2(C)CCC2)CCSC1)=O CS(=O)(=O)CC(=O)N1CCC(C(=O)NC2CCC(CO)CC2)O1 C1(CC=C)(C(=O)NC(CCNC(C)=O)Cc2cccs2)CC=CC1 CC(CO)C(=O)NCC(C)NC(=O)C(C)(C)c1cncs1 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(C)N(c2nnc(CO)s2)CC1 N1(C(c2c(N)csn2)=O)CC(NC(c2ccc3ccoc3c2)=O)C2CCCCC12 N1(C(C2(CNC(c3ccc(C)nn3)=O)CCCO2)=O)CCCC2(CCCC2)C1 C1(CNC(C=C(C)C)=O)CC2(CO1)CN(C(=O)Cc1ccc(CO)cc1)C2 C1(NC(C(C(C)C)CO)=O)CN(C(c2ncccc2F)=O)CCC12CCOCC2 c1(CC)oc(C(=O)NC(CNC(=O)C(CN(C)C)N(C)C)(CC)CC)cc1C N1(C(c2cnc(C)s2)=O)CC(NC(C23C=CC(CC2)C3)=O)C(O)C1 O=C1NCc2ccc(NC(C3CCC(NCc4cnc(O)nc4O)CC3)=O)cc21 c1(CC(=O)NCCNC(CN(C2CC2)CC)=O)ccc(Br)cc1C#N c1(C(=O)OC)cc(I)cnc1NC(C1CCN(Cc2ccccc2F)C1)=O CCC(CC(=O)N1CCCC(C)(C(=O)NCCOCCCCN=[N+]=[N-])C1)C(C)(C)C C(CN=C(NCC1COC(C)O1)NCC(C)(C)C)n1c(CC)ncc1 c1(OC)c(C)nc(N2CC(Cc3ccccc3)CC2=O)nc1C N(C1COc2ccc(F)cc21)C(c1cncc(N)n1)=O c1(C(N2CC(C)C(NC(=O)COC3COC3)CC2)=O)c[nH]c2cc(F)c(F)cc12 CC(C)(C(=O)NCC(O)CC(=O)N1CCC(N2CCC(O)C2)C1)C(F)(F)F C1(C2C(C(N(C3CN(C(C4CCN4C4CCCC4)=O)C3)C)=O)C2)CCCC1 C1(C(=O)NCc2n(C)cnc2)CC(O)C(O)CC1CNC(C1CC2(CC2)CO1)=O CC(CC(C)NC(c1cnoc1-c1cnn(C)c1)=O)NC(=O)C=CC1CCOC1 C1(NC(C2C(C)C2)=O)CN(C(=O)COCC2CCCCO2)CC2(CC2)C1 c1(NC(CC2N(C(C3CCN(C)C3)=O)CCCC2)=O)ccc(Br)c(F)c1F C1(C(=O)NCC2CC(C(NOCC(=O)OC)=O)C2)C2CCC(C2)C1C c1(C(N(CCCCCCNC(C2CC=CCC2)=O)C)=O)ccn2cccc2c1 N1(C(c2cccc(CC)n2)=O)CCN(C(=O)C(C)OCCOC)C2COCC12 C12(NC(C(C3CCCC3)OC)=O)CCCN(C(c3cncc(N)c3C)=O)CC1C2 c1(CC(=O)NC2CCCN(C(c3occc3Cl)=O)C2)cccc2nsnc12 Cc1cc2ncc(C(=O)NC(C)CN(C(=O)CC3CCCCC3(F)F)C)cn2n1 S(=O)(=O)(c1cnc(Cl)nc1)NC1CCN(C(c2cc3ccccc3o2)=O)CC1F c1(CC(=O)NCC2(NC(C(OC)OC)=O)CCC2)ccc(Cl)c([N+](=O)[O-])c1 O=C(C#CCNC(=O)C(F)C1CCCC1)NCCCn1ccnc1 C1(OC)CC(CNC(=O)CSCC2CCCO2)N(C(=O)Cc2ccncc2C)C1 C(N=c1[nH]c(C(F)(F)F)nc2cc(C(F)(F)F)ccc12)c1n(C(C)C)cnc1 N1(C(CCCC(=O)OCC)=O)CCCC2(NC(c3ccccc3)=O)CC2C1 CC(C)CC(C(=O)NCCC1(C)CC1(F)F)ONC(c1c(F)cncc1F)=O N1(C(c2c(OC)csc2)=O)CCc2sccc2C1CNC(C1(O)CC1)=O N1(C(CC(=C)C)=O)CCC2(CCN(C(=O)CCCC(C)CC)C2)C1 C(=O)(C(F)C(C)CNC(c1cn(CC)nc1C)=O)NC(CCC=C)C N1(C(C2(CCCC)CC2)=O)CC(NC(c2cc(C)cnn2)=O)CC(C)(C)C1 N1(C(c2csc(C(F)(F)F)c2)=O)CCCC1CC(=O)NC12CC(OC(C)C)(C1)C2 N(C(=NCC(C)COC)N1CCC(c2ccc(OCC)c(C)c2)C1)C(COC)C c1(OC)ccc(C(=O)NC2CC(NC(c3cccc(OC(C)C)c3)=O)C2)c(C)c1 C(N=c1nc(N2CC=C(C)CC2)c2c([nH]1)c(C)nn2C)c1n(CC)cnn1 CCCCCCC(C(=O)N1C2CCC1CN(C(c1cccn1C)=O)C2)NC(C)=O C1(N2CCCC2)(CC(=O)NC2CC(NC(C3CCSC3)=O)C2)COC1 CCCC(CNC(=O)COC(C)CC)C(=O)N1CC(CO)CC(C)C1 CCCC(C(=O)NCC1C2CC1N(C(c1ccn(CCOC)n1)=O)C2)C(C)C N(C1CC2(CCCC2)Oc2ccc(F)cc21)c1n(CC2CC(O)CC2O)nnn1 c1(C(N2CC(NC(C3CC(=O)NCC3)=O)C(O)C2)=O)ccc2ccsc2c1 CC1c2ncc(C(=O)Nc3cccc4c3OCO4)n2CCN1C(=O)CS(C)(=O)=O CC1=C(C(=O)NC(c2nn[nH]n2)c2cccs2)Cn2ncnc2N1C c1(C(N(C)CC2N(C(CCC)=O)CCCC2)=O)c(Br)ccc(C)c1C C(c1ccc(OC(F)F)cc1)=CC(=O)N(C1(N2CCOCC2=O)CC1)C1CC1 C1(NC(COCCOCC)=O)C(C)CCN(C(C2CC(=O)N2)=O)C1C C1(NC(c2c(C)nsc2C)=O)CN(C(=O)C2=NNC(=O)C2)CCC1C N1(CC(c2ccc(N(C)C)cc2)NCCCC(CC)O)C(=O)CC(C)(C)C1=O c1(C(N2CC(CNC(C=CC)=O)C(F)(F)C2)=O)n[nH]c2cc(Cl)ccc12 C1(CN(C(C2(F)CC2)=O)CC)CCN(C(C2CCC2(F)F)=O)CC1 Cc1nc2sccn2c1C(=O)NCC(F)CNC(=O)C1=NNC(C(F)(F)F)C1 C1(NC(CCn2cnc(=N)[nH]2)=O)C2CC3C1C3C2C(=O)NC(CCO)C(F)F N1(C(C=CCC)=O)CC2(CCCC(CNC(=O)NCCCl)O2)C1 c1(CC)cnn2ccc(C(=O)N(CCN(C(C3C4CC4C4CC34)=O)CC)CC)nc12 CCCCC(CNC(=O)CC1(C)CCCO1)NC(=O)Cc1csc(COCC)n1 N1(C(c2cc(C3CC3)no2)C(=O)N(C2(C)CC2)C2CCC2)CCC(O)(C2(C)N=N2)C1 C1(NC(c2ccc(F)cc2)=O)CCCN(C(=O)C=CCN2CCCC2)CC1 N1(C(C=Cc2cncc(C)c2)=O)CCN(C(=O)CC2(C)OCCO2)CC2(CC2)C1 c1(NC)cnccc1C(N1CCCC(N(C(=O)CC2CCCC(=O)N2)C)C1)=O Cc1nc(C(=O)NC2CCCN(C(C3CN(C4CCOC4)C3)=O)C2)c(=O)[nH]c1C C1(NC(c2n(C)ccn2)=O)CN(C(C2CNC(=O)C2)=O)CC1n1ccnn1 C(=O)(C1Cc2ccccc21)NC1CN(C(C2(NC(C)=O)CCCC2)=O)CC1O c1(C(C)NC(=O)CCOCCN(C(=O)CC2CC2)C)cn(C)nn1.C1(C)CS1 c1(N2CCC(CSC)C2)nc(=NCC(C)N2CCCCC2)[nH]c2c1CCCC2 N1(c2nc(C)c(C#N)cc2Cl)CCCC(C2CC2NC(=O)Cc2cc[nH]n2)C1 C1(NC(C2C(CCOC)C2)=O)CCC2(CC1)CN(C(=O)CC1(OC)CCC1)C2 O=S(=O)(c1ccc(Br)cc1N1CC2CCOC2C1)N1CCn2ncc(Cl)c2C1 C(CC(C)C)(C(=O)N1CCN(C(c2cnc(C)n2C(F)F)=O)CC1C)NC(C)=O N1(C(c2nc(C#C)sc2)=O)CCC(C(F)(F)F)C(NC(=O)CN2CC3CC3C2)C1 C1(O)(Cn2cc(C(C)N(C)C)nn2)CCN(C(=O)C(F)CC2CCCCC2)CC1 CCCC(C(=O)NCC(O)C1(Cl)CC1)NC(C1CCOC1C(C)C)=O c1(CC)noc(CC)c1CC(=O)NCCCC(C)NC(=O)CCCCSC Cc1nc(C)c(C(N2CC(NC(c3n[nH]c(C)c3O)=O)C(C)C2)=O)c(C)n1 c1(CC)ccc(C(=O)NC(C)C(=O)NCC2(C#N)CC2)[nH]1 c1(C(N2CCC(C3N(C(CCCC)=O)CCCC3)C2)=O)cc(CCOC)nc(O)c1 C(=O)(C1COc2ccccc21)NC1C(NC(c2cc(C)[nH]c2C)=O)COC1 N(C1CCc2cccc3cccc1c23)C(C(=O)N(C)CC)=O c1(N(CCCNS(C)(=O)=O)C)nc(N(C)CC2(F)CC2)nc2ccsc12 CCC(C)(C(=O)N1CCC(OC)C1)NC(c1ccc(-c2ccc(C)s2)s1)=O c1(C(=O)NC2CCC(C(N(C3(CO)CC3)C)=O)CC2)cnccc1C#N Cc1nn(C)cc1CNC(=O)CCc1ccc(C(=O)NCc2cccc(Cl)n2)[nH]1 N1(C(c2c(CC)n[nH]c2)=O)CCN(C(=O)CCc2cnn[nH]2)C(C)C1C N1(CC(=O)Nc2ccc(CC)cn2)CCC2CCC(C2)C1.C12CC(C1)C(=O)N2 c1(CC(N2C(C)(CNC(CCOC)=O)CCC2)=O)cccc(F)c1Cl C1(NC(C2OCCC(C)C2)=O)CC1C1CCN(C(c2cc(C3CC3)on2)=O)CC1 C1(NC(c2cnc(C(C)O)s2)=O)CCC(CN(C)C(C2CC(Cl)(Cl)C2)=O)CC1 C(=O)(C(C)(F)C(C)(C)F)NC(CC)CNC(=O)C(C(C)C)NC(C)=O c1(CN(C(CC#C)C)C(c2ccc(OC(F)F)cc2)CC)ccccc1OC Cc1cc(CC(=O)NC(CNC(=O)CSC2CC2)C2CC2)ccc1O C1(CC=C)(NC(=O)CCCOC(C)C)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1 O=C1CC2(CCN(C(C3CC34CCNC4)=O)C2)CN1 C1(CCNC(CSCC#C)=O)CN(C(c2cc(N)cnc2C)=O)CCS1(=O)=O c1(C(N2CCN(C(C3CCCC3)=O)C(CO)C2)=O)nc2cccnc2s1 N1(C(C2C(C)C2)=O)CCC(O)(CCNC(=O)CN2CCC(C)(C)C2)CC1 n1(CCC(=O)OCC)cc(CCNC(=O)CC2C=CC(NC)C2)nn1 N1(C(c2c(C)cc(CC)o2)=O)CC(NC(=O)C(n2ccnc2C)C)CC(C)C1 c1(NCC=CC)cc(S(=O)(=O)NC2(c3ccccc3)CCC2)ccc1C#N CN1CCN(C(=O)Cc2nc(=N)[nH][nH]2)CC1C(N1CC(F)C1)=O Nc1c(Cl)cc(C(=O)NCC(F)CNC(C2CC2C2CC2)=O)cc1[N+](=O)[O-] C1(CNC(C(C)OCC#C)=O)CC(CNC(c2csc(C(C)C)n2)=O)CO1 c1(C(=O)NC2C(NC(CCCN(C(C)=O)C)=O)COC2)cc(C(C)(C)C)nn1C C(CC(=O)C(C)(C)C)N(CCCc1cnoc1)C c1(CN(C)C(C2(C)CC3CC3C2)=O)cc2cccc(F)c2s1 c1(C(C(N2C(CNC(c3c(CC)cco3)=O)CC2)=O)C)ccccc1Cl N1(C(C2CCC(N(C)C)C2)=O)CCN(C)CC1CNC(=O)C(C)(C)n1cnnn1 C1(C(=O)NC(CC)CSC)(OC)CCN(C(c2coc(Cl)n2)=O)CC1 c1(C(CSCC(=O)NCC(C)N(C(=O)CCn2cncn2)C)=O)ccccc1 C(=O)(C(CC#CC)NC(c1ccc(F)c(F)c1)=O)N1C(CCC#C)CCC1 CC1(C)CCCCC1(C)NC(C1C(C2CC2)CCN1C(=O)CN1CCCCC1)=O C1(NC(COCC(=C)C)=O)COC2(CCN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)C1 c12cccc3c1nnn3C(CC)C(Cl)(C(=O)OC)CCNC2=O c1(OC)ccc(CC(=O)NC2(CNC(C3CC3(C)Br)=O)CCCCC2C)c(Cl)c1 c1(C(N2CCC3(C(NC(COC4(C)CCC4)=O)C3)C2)=O)cc2ccsc2n1C c1(CC(N2CCN(C(CCC=CC)=O)CC2C(C)C)=O)c(F)cccc1C#N CC(O)(CNC(=O)C=CCNC(=O)COC1CCCC1)CO c1(OC)ccnc(C(N2CCC(O)(CNC(C3(C)C=CCC3)=O)C2)=O)c1OC Cc1ncnc(C(=O)NCC(C2CCC2)NC(c2cccc(N(C)C)c2)=O)c1C c1(CCC)onc(C)c1C(N1CC(NC(C2C=CC=CC=C2)=O)C(C)C1)=O C(=O)(CC(F)(F)C(C)C)N1CCC(N(C(C2CC(OC)C2)=O)C)C1 c1(N(C2CCCC2)CC#C)nnc(C2CC(O)C2)n1CC1CCN(C)C1 c1(CC)ncc(C(=O)N(C2CCC(NC(C3(Br)CC3)=O)CC2)C)c(C)n1 C(CCN=c1[nH]c(Cl)ncc1C)OCCNC(c1c2cccc(C)c2sc1)=O c1(C(=O)NCC2CN(C(C3CCCCC3)=O)CCO2)cc2c(O)ncnc2cn1 c1(OC)ccc2c(c1)CC(C)N2C(=O)NC(c1ccoc1)C C1(C#N)(C(c2n(CC=C)nnn2)NCc2ncc(Cl)n2C)CCCCC1 c1(C(N2CCC(OC)(CNC(=O)CCS(C)=O)C2)=O)cncc(F)c1Cl N1(C(c2c(OC)ccs2)=O)CCCCC(NC(=O)CC2CC(OC)C2)C1 C1(CNC(C(CC)(C)C)=O)CC2(CCN(C(=O)CC3CCNC3=O)CC2)CO1 c1(C(=O)OCC)ccc(NC(=O)CCCn2ccnn2)cc1.C1(CNC=O)(SC)CC1 C#CCC(C(=O)NCC1(O)CCN(C(c2ccc(C(C)C)s2)=O)C1)C1CC1 c1(SC)ccc(CNC(C2CSCCN2C(C2(O)CC2)=O)=O)cc1 C(=O)(C#CC1(C)CCCO1)N1CCN(C(c2cncc3c2CCC3)=O)CC(C)C1 C1(N(C(=O)CSCc2ccccc2)C)CC2CCC(C1)N2C(=O)CC1(CO)CC1 c1(C(=O)NCC(C)CN(C)C(c2ccco2)=O)cc(S(N)(=O)=O)ccn1 c1(CN2CC(F)(C(N3CCCC3)=O)C2)nc(Br)ccc1F n1(CC)c(C(N2CCC(NC(=O)C(C)(Cl)Cl)C23CCCC3)=O)cc2ccccc12 Cc1c(CC2(NC(=O)NC3CCN(C)C3c3cccnc3)CC2)cccc1Br N1(C(c2cc(C)c(C(N3CC4CC3CN4C)=O)o2)=O)CCC2(CC1)CC2CO C=CC(CC)C(=O)NCCOC(C)(C)CNC(=O)C(CO)NC(N)=O C(=O)(C(O)CC(F)F)N1CCCC(N(CCNC(C)=O)C)C1 c1(OC)cc(OC)c(C(N2CC(NC(C3CC(C)(C)CO3)=O)C(O)C2)=O)cc1N CN1C(=O)CCC1C(=O)NCCCCNC(=O)CCn1ccnc1 C12(CF)COC(C(NCC)=O)(C1)C2.C1(C(C(=O)N(CCN)CC)OC)CCCCC1 C1(NC(c2cc(C(N)=O)[nH]c2)=O)CC2CC(NC(=O)CCc3cncnc3)C2C1 Cc1ncnc(C)c1C(=O)Nc1cccc(CC(=O)NC2CCS(=O)(=O)C2)c1 Cc1onc(C(=O)N(CC(C)CNC(C2CC2C(C)(C)C)=O)C)c1Br C#Cc1cnn(CC(=O)NCC(c2ccc(F)cc2)NC(=O)C(COC)SC)c1 N1(C(CCC=CCC=C)=O)C(C(=O)NCC2CC2[N+](=O)[O-])CC2CCCC12 N1(CCNC(C2CN(C(=O)Cc3cncc(O)c3)C2)=O)CC2CCC1C2 CC(C(=O)NCC1CC1CNC(c1ccc(C2(C)CC2)cc1)=O)C(C)(C)C c1(C(=O)NC(C(C)C)(C)CNC(c2cc(Cl)ns2)=O)ccc2nncn2c1 C(=O)(C(O)C(F)F)NCC(C)(C)NC(=O)CCc1ccc(O)cc1 c1(C(C)NC(=O)COCCCCCN(C(=O)C=CCO)C)ccccc1 c1(C(=O)NCC2CC(NCc3ccc(OC)c(CO)c3)C2)ccc(C#N)c(F)c1 C(C)(CNC(=O)CSc1cn[nH]c1)(CC(C)C)NC(C(CSC)C)=O C1(N(C(=O)NC2C(C(C)(F)F)C2)CCN)CCCCNC1=O.c1(OC)ccccc1Br c1(C(C(=O)NCCCOC)N(C)Cc2cncn2C)nc(Cl)sc1Cl C1(C(C(C)C)NC(CSCC)=O)CCN(C(=O)CCc2ccccc2Br)CC1 N1(C(C2C(C)(Br)C2)=O)CCCCC12CC(NC(c1ccc[n+]([O-])c1)=O)C2 C12(NC(c3c(C)cno3)=O)CCCC1N(C(c1nn(C)cc1Cl)=O)CCC2 O=C(C1=C(Cl)CCOC1)N1CCC1CNC(C12CCC(CC1)O2)=O c1(C(N2C(CNC(C3C4COCC34)=O)CC(OC)C2)=O)cc2c(=O)cc[nH]c2s1 C12(C(=O)NC(c3n(CC)ncc3)C)C(NC(C3CCC(=O)N3C)=O)C3CC1C2C3 C1(C(=O)NC(C2CCCCC2)C)CCN(C(=O)C(n2cc(Cl)cn2)C)CC1O C12(C(N3CC(O)(CNC(c4nccc(C)c4N)=O)C3)=O)CC3CC(C(=O)N1)C2C3 C1(N(C(=O)NC(C2CCOC2)C)C)CCN(c2ccccc2)CC1 NS(=O)(=O)c1cccc(NC(=O)NC2CC(F)CN2C(=O)C2=COCCO2)c1 C(C)(CC(C)N=c1ccnc(SC)[nH]1)NC(c1ccc(N(CCC)CC)cc1)=O c1(OC)c(F)cc(C(=O)NC2C3CC(O)C2N(C(=O)C2CC2)C3)cc1Cl N1(C(=O)COCc2cccnc2)CCN(C(C2CC3(C2)CC(O)C3)=O)C2CC12 N1(C(CS(CC)=O)=O)CCC2OCCN(C(C3(C(=O)N(C)C)CC3)=O)C2C1 c1(C(N2CC(NC(c3cc(SC)oc3)=O)C(F)C2)=O)cc2ccccc2cc1Cl N1(C(=O)Nc2ccc(SC)nc2)CC2(CCCC2NC(=O)NC(C)(C)C)C1 CCCCC(C)(F)C(=O)N1CC(NC(c2ncnc(C(F)F)c2OC)=O)C1 c1(C(=O)NC(CNC(CCCC=C)=O)C)cc(Br)cc([N+](=O)[O-])c1Cl N1(C(c2cc3ccncc3s2)=O)CCCCC(N=c2ccc3nnnn3[nH]2)C1 C(=O)(CC(C)(C)CC(F)F)NC1CN(C(C2(C)CN(C)C(=O)C2)=O)CC1N=[N+]=[N-] c1(C(N2CCC(NC(CCNC(CC(C)C)=O)=O)C2C)=O)c(Br)c(C)nn1C N1(CCN(C)C(c2csc(O)n2)=O)CCN(C(=O)C(F)C2CCCC2)CC1 C1(CNC(C2(OCC)CCC2)=O)CC(NC(c2ccc(O)nc2)=O)C(O)C1 C(C(=O)NCCC1(C(=O)NC2CC(F)C2)CC1)(C(C)C)OC CC1CC(NC(=O)C(F)(Cl)c2ccccc2)CN(C(c2sccc2Cl)=O)C1 c1(C(N(C)CC2CCCN2C(=O)CSc2nncs2)=O)ccn2nncc2c1 C1(CCC(N2CCC(OC)C2)=O)CN(C(C2CC2C(=O)OC(C)(C)C)=O)CCO1 N1(C(C(CC)NC(=O)CN(C)C)=O)CC2CCN(C(=O)CCSC)CC12 CC1CC(N=c2[nH]c3c(c(=NCc4ncn(C)n4)[nH]2)CCCCC3)C1 N1(C(C2N(CC)CCC2)=O)CC2CC1CN2C(c1ccc(C(F)(F)F)nc1)=O CC1CCCCC1(CNc1ncc(C(C)(C)O)cn1)NC(C1COC(C)(C)C1)=O C1(C(=O)NCCC(C)(C)NC(C2C(c3n(C)nnn3)CCC2)=O)CCC2(CCC2)O1 N1(C(C2N(Cc3ccn(CC)n3)CCC2O)=O)CCC2(CC1)CN(C)C2 c1(C(N2CC(NC(c3cnc(Br)o3)=O)C(F)C2)=O)cccc2cc(O)ccc12 c1(OC)ccc(CC(=O)O)cc1S(=O)(=O)N(Cc1ccccc1)C.C(=O)(C(N)=O)N c1(C(=O)NC2(CNC(C(c3cnn(C)c3)C)=O)CCC2)ccc(N)cc1Cl C1(C(=O)N(C2CC(CCC(=O)OCCO)C2)C(C2CCOC2)C2CC2)CCC(=O)O1 C1(CNC(C2CCN(C(C)=O)C2)=O)(CO)CCN(C(=O)Cn2cccn2)C1 C1(CC(=O)NCC(C2CC2)NC(=O)Cc2cccc(Cl)c2)CC2(CCC2)C1 N1(C(c2ccn(C)c2)=O)C2CCC1CN(C(=O)CC1CCCCC1(C)C)C2 C#CCC(CC(=O)N1CCC1C1CCCCC1)NC(C1(C)COC(=O)N1)=O CC1=C(C(=O)NCC2(NC(c3cc(C)cs3)=O)CCCCC2)CCCO1 c1(CSCCC(=O)N(CCCCCNC(C2(C#N)CC2)=O)C)ccc(F)cc1 C(CCCCC(=O)N(C1(C)CCS(=O)(=O)C1)CC(=O)O)SC C1(NC(CC(CCC)O)=O)CN(C(c2ccc(C)s2)=O)C2(CCCCC2)C1 CCC1=C(C(=O)NCC2(n3cccn3)CCN(C(C3CC3=C)=O)CC2)SCCO1 N1(C(CC=C(C)C)=O)CC2CCC1C1CN(C(c3cnnc(O)c3)=O)CC21 c1(N(C2CN(C(C(=Cc3cn[nH]c3)C)=O)C2)CC(C)O)ccc(F)c(F)c1 Cc1ccc(C(F)(F)F)cc1C(N1CCC(O)(CNC(c2csnc2C)=O)C1)=O c1(NC(C(C)N(C(C(CCCC)C)=O)C2CCC2)=O)cnc2ncnn2c1 N1(C(c2cc(Br)c(C)cn2)C(=O)NC(CC)C)C2CCCC1CC(N=[N+]=[N-])C2 CC1(C)Nc2ccccc2C1NC(c1ccccc1C(F)(F)C(F)F)=O Cc1cn2ccc(C(N3CCC(CN(C)C(c4cncnc4)=O)CC3)=O)cc2n1 C1(C)(CC)CC(C(=O)NCC(C2CCCC2)NC(C2CCCO2)=O)CCO1 Cc1[nH]cc(C(=O)N(C(C)CCNC(=O)CC2CCCCCO2)C)c(=O)c1Cl CS(=O)(=NC(=O)C1CCC2(COCCO2)O1)C1CC(CN)C1 CCCC(CCCNC(c1cnc(S)n1C1CC1)=O)NC(C1CCCNC1=O)=O c1(C(N2CCN(Cc3cnc(CCC)o3)CC2)=O)cc2c(Cl)cccc2nc1C c1(CC(C(=O)OCC)NC(c2ccc(C#N)cc2)=O)c[nH]c2cnccc12 C1(C(=O)NC2CN(C(Cn3nc(C4CC4)n(C)c3=O)=O)C2)CNC(=O)CC1(C)C C1(C(N2CCC(CNC(C3SC4C=CC3CC4)=O)C2)=O)CC2CS(=O)(=O)CC2C1 O=C(C1OCCc2ccc(Br)cc21)N1CC(C2CC2)(c2nn[nH]n2)C1 c1(OC)cc(C(N)C(=O)NC2(c3ccccc3)CC2)cc(OC)c1OC C(=O)(C(Cc1cn[nH]c1)NC(c1cc(C)no1)=O)NC(CCC)C1CC1 C(=O)(C1=CCN(C(C2(CO)COC2)=O)C1)NC1C(C)(C)C(O)C1 c1(C(N2CC(C)(CCC(=O)NC(C)CO)C2)=O)ccc(C#N)cn1 C1(NC(=O)CC2COCCO2)COC2(C1)CN(C(c1ccc(O)c(F)c1)=O)C2 C(C)(C(C)S(C)(=O)=O)NC(CC(=O)OC)(C)c1ccccc1.c12ccc(o1)s2 c1(OC(c2ccccc2)COC)ccccc1NC(=O)Nc1ccccc1Cl CCC(CN=C(NC1CCCC1)N1CCC2(C1)CC2(F)F)C(F)(F)F C1(NC(C2(C(=O)OCC)CCC2)=O)CS(=O)(=O)CC1NC(c1cc(C)[nH]n1)=O C1(C(N(C)CCNC(c2cccc(N3CCCC3)n2)=O)=O)CS(=O)(=O)CCO1 Cc1nnc(C(C)(C)NC(C2CC2C(C)(C)C)=O)s1.c12c[nH]nc1CCNC2=O C1(C(N2CC(N(C)CC)C2)=O)CN(C(=O)COCC2CCCO2)CC1(C)C N1(C(COCCC(C)C)=O)CCC2(CC(NC(=O)CC3CCCC34CC4)C2)C1 c1(C(=O)NC2(CNC(C3N(C)CCC3)=O)CCCC2)cnc(Br)c(N)c1 N#Cc1cncc(C(N2CCCN(C(c3ccc(Br)nc3)=O)CC2)=O)c1 C=CC(O)C(=O)NCC1CC(NC(C2(Cc3ccccc3)CC2)=O)C1 c1(OCC)cccc(CC(=O)NCC2CN(C(=O)C=C(C)Cl)C3CC23)c1 C1(NC(c2cn(CCC)nn2)=O)CCCCC1CNC(C1(C)CC2CC2C1)=O N1(C(CCOCC#C)=O)CSCC1C(=O)NC(c1nncn1C)C c1(OC)cc(C(=O)NCCn2cccn2)c(NCc2cccc(F)c2F)cn1 c1(C(C(=O)NCCC2(NC(CCC3C(C)(C)C3)=O)CCC2)C2CC2)ccccc1 C(=O)(C(CNC(=O)C(c1cn(C)nc1C)C)C(C)(C)C)NCCOCCCC#C C(=O)(CC(C)NC(c1c[nH]c(=N)o1)=O)NCC(n1ccnn1)C CC1CCOC(C(N2CC(O)(CCNC(=O)C(c3cnn(C)c3)O)C2)=O)C1 C1(NC(c2cc(C)oc2C)=O)CC1C1CCN(C(=O)C(C2CC2)N(C)C)CC1 c1(C(N(C2CC2)CC2CCN(C(C(N)=O)=O)CC2)=O)ccc2cccnc2c1 c1(C(=O)NCC2CN(C(c3cc(Cl)cs3)=O)CCO2)ccc2ncsc2c1 C(N=c1cc(C2CC2)nc(Cl)[nH]1)C1CCN(C(C(C)(C)CF)=O)C1 N1(C(C2CCCS2(=O)=O)=O)CCC2(CCN(Cc3cccc(Cl)c3[N+](=O)[O-])C2)C1 N1(C(C(C)OCC)=O)CCCC(C2CCN(C(C3(C(F)F)CC4(CC4)C3)=O)C2)C1 C1(C)(CNC(C(C(C)C)c2cccnc2)=O)COCCN(C(=O)C(C#N)C2CC2)C1 C1(C(N(C(C2CCCNC2)C)Cc2scc(C)n2)=O)CC2CCC1CC2(C)O c1(C(c2nnnn2C(C)C)NCC2CC(CO)C2)cc[nH]c1-c1ccccc1 CP(C)(=O)C1CCCCN1C(=O)C(CCC(N)=O)n1cc(C2(O)CCCC2)nn1 N1(C(c2cnn(C)c2N)=O)CC(NC(c2csc(C3CC3)n2)=O)CC(C)(C)C1 Cc1nc(Cl)cc(Cl)c1C(N1C2CC1CN(C(=O)CC1CCCC1)C2)=O N1(C(c2ccc(OC)cn2)=O)CC2CCC(C1)N2C(C1(C(F)(F)F)CCC1)=O N1(C(C(CN(C)C)NC(C(C(C)O)N(C)C)=O)=O)CCC12CC(O)C2 c1(C(=O)NC(CC(F)F)C(=O)N2CCOC(C3CCC3)C2)nccc2[nH]ccc12 Cc1cc(C(=O)NC23CCOC(CNC(=O)C(C)O)(C2)C3)c2c(c1)CCO2 c1(C(N2CC(CNC(C3CCCC3)=O)OCCC2)=O)cc(F)c(O)c(F)c1 C1(C(N(CC(C)(C)CNC(=O)CCc2ccc(CO)o2)C)=O)CCCC(C#N)C1 c1(C(=O)NCCCn2cc(CNS(C)(=O)=O)nn2)ccc(-c2ccco2)nc1 CCC(CCCC(=O)N1CCCCC1C(F)F)NC(C1CCN(CC)C1)=O c1(C(CNC(c2snnc2C2CC2)=O)O)cccc(Cl)c1Cl CCC(CC)CC(F)C(=O)NCCSC.C1(=O)C(C(=O)OC)OC(=O)C(C)N1C CC(O)(CC(=O)NCC1(C(N)=O)CN(C(C2(c3cc[nH]n3)CC2)=O)C1)C1CC1 Nc1cc2c(cc1C(N1CCOC(CNC(=O)Cc3cccs3)C1)=O)OCO2 C1(C(N2C(C)CC(NC(c3csc(C(F)F)c3)=O)CC2)=O)CCC2CC1C2(C)C CN1CC(C(=O)NC2CC23CC(NC(c2ccc(OC(F)F)nn2)=O)C3)CC1=O C1(SC)CCN(C(C2CCC2CNC(=O)COCC2CC2)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC3)=O)C2)cc(=O)cc[nH]1 c1(OC)c(C(=O)OC(C)C(=O)NO)cc(Cl)cc1C c1(CC(=O)N(CC(C)O)CCNC(c2sccc2C(F)F)=O)ccccc1Cl C1(CC)CN(C(c2cc(C)nc(C)c2)=O)CCC1CNC(=O)C(O)C(F)(F)F C1(NC(Cc2nc(C)oc2)=O)CN(C(=O)C(O)c2ccco2)CC1C1CC1 C(C)(C(=O)NOCc1ccsc1)NC(C(C)CC1CCCC1)=O Cc1cc2c(C(=O)NCCCCNC(c3cc(CO)c(C)o3)=O)nccn2n1 Cc1ncc(Cl)c(C(=O)NCC(Cc2ccccc2)NC(=O)C=CBr)n1 C1(CCC(=O)NC(CNC(COCCCC)=O)CC)CCCCN1C c1(Oc2ccc(NC(=O)Nc3csnn3)cc2)ccc(Cl)cc1Cl c1(CN=C(NCc2c(COC)noc2)NCc2ccc(Cl)cn2)cccc(OC)c1 C1(C(=O)NCCNC(=O)CO)CCCC1NC(=O)C=C1CCOCC1 n1(CC(N2CC(NC(COCCOC)=O)C(C)CC2)=O)cnc2sccc2c1=O C12COCCC1NC2=O.c1(C(N)=O)cc(NC(c2cc(COC)on2)=O)cnn1 CCC(COC)(CC)C(=O)N(CC(O)CNC(c1cnc(C)[nH]c1=N)=O)C N1(C(CNC(CC)=O)=O)CCOC(CC(N2CCC(F)(CF)C2)=O)C1 N1(C(C2(C)CC(F)C2)=O)CC(Nc2cc(O)ncn2)CC2(CCC2)C1 c1(CC(=O)NCCN(C(c2c(CC)non2)=O)C2CC2)cccc(OCCC)c1 C1(CCNC(CC2(C(C)(C)C)CC2)=O)CN(C(C2CC3CC3C2)=O)CCS1(=O)=O c1(C(N(C2CN(C(C(C)Oc3ccccc3)=O)C2)C)=O)cc(N)ccc1CO C12(C(N3CCC(NC(CC(CC)C)=O)C(O)C3)=O)CCC(CC1)C(C)(C)O2 CC1CCC(NC(=O)COc2ccc(Cl)cc2)CN1C(c1csc2nccn12)=O N1(C(CCCC2C(C)C2)=O)C(C(=O)NC2CC3CCC2C3)CCC12CC2 Cc1nc(=NC(CNC(c2cccc(C#N)c2C)=O)CO)s[nH]1 N1(S(C(CC)C)(=O)=O)C2CCC1CC(NC(c1ccc(OCOC)cc1F)=O)C2 CC1CCN(C(=O)CC2(O)CCCOC2)C1CNC(=O)Cc1cncnc1O N1(C(C(C)(C2CC2)OC)=O)CC2C(CNC(C3CCC4(CCC4)C3)=O)C2C1 c1(OC)cncc(C(=O)NC2CCCC(N(C)C(c3cc(C)ncn3)=O)C2)n1 N1(CCN(C(c2cc(C)no2)=O)C)CCN(C(=O)CSC(F)F)CC1 CON=CC(=O)NCCC1CCC(NC(C2CC(CC(F)(F)F)C2)=O)C1 C1(CNC(N(C=O)Cc2nc(CC)sc2)=O)CC12CCS(=O)(=O)CC2 n1(CC(=O)NC2C(CNC(c3c(CC)con3)=O)CCC2)cc(C#N)cn1 CC(C)C(C)(O)C(=O)NC1CC(O)C1CC(N1CCC(O)(CO)CC1)=O C1(CC)(CC)CCCN(C(C2(NC(C3CCN(C)C3=O)=O)CC(F)(F)C2)=O)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)N1CC(C)C(CCNC(=O)CC23CCCC2C3)C1 Cc1ccc(C(N2CCCC(N(C(=O)CCC3CCOC3)C)CC2)=O)cc1C N1(C(c2ncc(OC)cc2F)=O)CCC2(CCCCN2C)C1 C1(OC)C(COC(c2cccnc2)=O)CN(C(=O)C(OC)OC)C1CO N1(C(C2C(OC)CCC2)=O)CCCC(C)C1CNC(c1ccnc(F)c1)=O CC1=CCN(C(=O)C(c2ccccc2)NC(C2CN(C(N)=O)C2)=O)CC1 C1(C(N2CCC(O)(C(C)NC(=O)C=C3CCC3)C2)=O)CN(CP(C)(C)=O)C1 c1(CC)cnccc1C(=O)OC(C)C(c1cccn1C)=O C1(C(N2CCCC(c3cn(CCC=C=C)nn3)C2)=O)CC2CCC(C1)O2 c1(C(=O)NCCNC(c2cc(CCC)on2)=O)ccc2c(=N)[nH]cnc2c1 c1(-n2c(C(O)C3CC3)nc(CC)n2)ccc(F)cc1OC c1(C(=O)NCC2(CNC(c3cc(C)n(C)c3)=O)CC2(F)F)ncc(N)cc1Cl C#Cc1cnn(C)c1C(=O)NCC1CC1CNC(C1(CC2CC2)CCC1)=O C12(NC(C3CCN(CC(C)C)C3)=O)COC(C1)C(NC(c1ccn(C)c1)=O)C2 c1(C(=O)NC)ccc(NC(C2CC23CN(Cc2c(Br)cnn2C)C3)=O)cc1 CCCCCCCC(=O)NC(C)(CO)C(=O)NCCCn1cncn1 c1(C(=O)OC)cnc(C(=O)Nc2cccc(CO)n2)cn1 CC(C)C(CCC(=O)NOCC1CC1)NC(c1ccc(O)cn1)=O N1(C(C2CN(C(N)=O)C2)=O)C2CCC1CN(C(C1Cc3nncn3C1)=O)C2 NS(=O)(=O)C1(C(=O)NC2CCC(NC(=O)CCc3ccc(O)nc3)C2)CC1 C1(NC(c2c(=N)[nH]cnc2)=O)C2CCC1N(C(c1cccc(C3CCC3)c1)=O)C2 C(=O)(C1CCCc2ccnn21)NCC1CN(C(CCCN(C(C)=O)C)=O)CC1C N1(CC(=O)N(CC(CNC(C2(C(C)O)CC2)=O)C)C)CCc2sccc2C1 c1(C(C(=O)NCCCNC(=O)NC)NC(=O)C(O)c2ccsc2)cccnc1 c1(C(=O)NC2C(CC)N(C(=O)CCOC(C)=O)CC2)cccc2c1OCC2 Cc1ccc(CC(=O)N(CCCOCCNC(C2(C)CC2(F)F)=O)C)cc1O C1(CC2N(C(C)=O)CCC2)CCN(C(c2coc(C3CCCCC3)n2)=O)CC1 CC1CN(Cc2ccc([N+](=O)[O-])cc2)CCCC1Nc1cscn1 N1(C(c2cnc(CSc3c(C(=O)OC)cn(C)n3)s2)=O)CCC(C(F)(F)F)C1C c1(C(c2nnnn2CCCOCC2CC2)NC(C)CCO)c(Br)ncn1C N#Cc1ccncc1C(=O)NC1CC1C(=O)Nc1cccc(C2CC2)n1 N1(CC(=O)NCC(C)(C2CC2)NC(C(C)N(CC(F)(F)F)C)=O)CCCCC1=O c1(C(=O)NCC(CNC(=O)CN2CCC(O)CC2)F)cnn2c1CCC2 c1(N2CCCC(CNC(C3(CC(C)C)COC3)=O)C2)nc(Cl)ncc1[N+](=O)[O-] c1(C(=O)NC2(CC=C)CN(C(=O)C=Cc3cccnc3)C2)ccc(CSC)cn1 c1(C(=O)NC2CC(NC(C(C=C)O)=O)CC2O)oc2ccccc2c1Br C1(CNC(CCc2ccc(C)cc2)=O)CC2CC1CN2C(=O)Cn1nnc(=O)[nH]1 N1(C(C2C(CC)C2)=O)CC(N(C(=O)CNC(=O)COc2ccccc2)C)C(O)C1 CCCC(C(=O)N1CCC1)N.C1(OCCOC)CCN(C(=O)C(=O)NC)CC1 C1(NC(C(c2scc(C)n2)C)=O)CCN(C(c2cn(C(C)C)nc2C)=O)C(C)C1 N1(C(Cc2c(C)nsc2)=O)CCOC(C(C)NC(=O)COc2ccsn2)C1 C1(C(N2CCCC(N(C(C3(C=C)CCC3)=O)C)CC2)=O)CN2CCCCC2CO1 N1(C(=O)CC2CC(F)(F)C2)CC2CCCC(C1)N(C(=O)CC1CCOC1)C2 c1(OC)cc(N2C3CCC2CCC3)cc(CN(CCO)CCO)n1 C12(COC)CC(NC(=O)C=C(C)C)(C1)C(C)O2.C12CC(C1)CNC(=O)C(=O)N2 C1(C(=O)NC(CC=CC)C(=O)N2CC3(CSC3)C2)CCCC(C)(C)C1 c1(CC(CC)C)nc(CC(O)C2CC2)n(-c2cn[nH]c2)n1 N1(C(c2cn(CC)nn2)=O)CC(C)C12CCOCC2.C(C(C)C(=O)N(CCOCC)CC)O N1(C(c2cc(C)n(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])n2C)=O)CC(CO)C1 C12(NC(CSCC(=O)OC)=O)CCC(NC(C3COCCN3C)=O)(CC1)C2 C#Cc1cnc(C(N2CCCC2CNC(=O)COCC)=O)c(C)c1.CC=C NS(=O)(=O)c1ccc(CC(N2CC3CC2C3NC(=O)C(O)CC(F)(F)F)=O)cc1 C=C(C)C(CC(=O)NC(C)CN1CCCC1)OC.C1(=O)CCNC(=O)NCCN1 c1(C(=O)NC2C(NC(C(C)=C(CC)C)=O)CCC2)cccc(NC(N)=O)c1 Cc1ncccc1C=CC(=O)NCC(C)NC(C1(O)CCCCC1)=O.C(CO)S C1(NC(CCOC)=O)CCC(C)(C)CC1CNC(=O)C(=Cc1c[nH]cn1)F C1(C(N2CC3C(CNC(=O)Cn4cc(Br)cn4)(C3)C2)=O)CCCC(F)(F)C1 c1(C(=O)NCC(C)(C)NC(C2CN3CCN2CC3)=O)ccc(Cl)c(N)c1 N1(C(Cc2c(C)ocn2)=O)CC2(CNC(c3c(O)cccc3F)=O)CCC1CC2 CC1CC(C(=O)NCC2CCCC23CC3)N(C(c2cn(CCO)nn2)=O)C1 CC(C)CCC(O)C(=O)NCC(CC1CC1)C(=O)NC1(C2CCCO2)CC1 O=C(C(O)CCNC(C1CC2CCC1O2)=O)NC1CC(n2cncn2)C1 c1(C(C(=O)NC2COC2)N(C2CC2)CC)cn(CC2CC2)nn1 Cc1cc(C)c2nc(N3CCC(C)C3CNC(c3ncccc3CO)=O)sc2c1 C1(C)(CNC(C2(CC)CCC2)=O)CCC(NC(=O)Cc2ccccc2F)C1 Cc1cc(C(=O)N(C)CCN(C(=O)C(CO)NC(=O)C(C)C)C(C)C)cn1C N1(C(C(CC2CCC2)OC)=O)CC(C(=O)NC2CC2c2ncccn2)C2(CC2)C1 N1(C(C2CCN(C)C2=O)=O)CCC(C2CN(C(C3CC=CCO3)=O)C2)CC1 c1(C(=O)NCC2CN(C(C(C)CF)=O)CC2C(F)(F)F)cc(N)cc(F)c1 c1(OC)cc(CCCNC(=O)NCC(C(=O)O)C2CCOC2)ccc1Cl N1(C(C(C(C(C)C)O)C)=O)CC2CCN(C(c3nnsc3N)=O)CC2C1 c1(C(N2CCC(OC)(CO)C2)=O)cc2n(c1)CCNC2 c1(CCC=C)ccc(C(=O)N(C2CN(C(=O)CC3CC3)CC2O)C)cc1 CC(C)(C(=O)NCCC1COCCN1C(C1OC2CCC1C2)=O)C(F)(F)F C(CC(=O)NCC1CC2(CCCC2)C1)(C(C)CC)NC(CCC=CCC=C)=O c1(N2CCC(SC)C2)nc(=NCCC(C)c2ccccc2)[nH]c2ccsc12 C1(C(C)C)C(C(C)C)CN1C(=O)C(N1CCOCC1)C C1(NC(CCC(=O)N(CCC)CCC)=O)CN(C(=O)C2=CCOCC2)CCC1CO c1(C(CC)=O)ccc(NC(=O)CN(C)CC)cc1.C12CN(CC1O)CC(=O)N2 N1(C(C(CC)=CC)=O)CCCC2(C1)C(NC(=O)CC(O)CN(C)C)CCN2C C1(NC(=O)COCC2CCCOC2)CN(C(c2cnc(S)[nH]2)=O)CC12CC2 c1(C(=O)NC2CC3(CCN(C(CC4CC(=O)C4)=O)C3)C2)ccc2nc(O)[nH]c2c1 CC(C)C(N=c1[nH]nc(C#N)s1)C(C)NC(=O)Cn1nnc2c1CCC(CO)C2 C1(c2n(CC(=C)C)nnn2)(NCc2cc(Br)no2)CC2CCCC12 CC(O)(Cn1cccn1)C(=O)NCC(C1CC1)NC(c1ncccc1Br)=O N1(C(CNC(C)=O)=O)CCOC2(CCC(NC(=O)Cc3c(C)noc3Cl)CC2)C1 C1(NC(CC2CC(=O)NC2=O)=O)CCN(C(c2cc(CO)[nH]n2)=O)CCC1CO c1(C(=O)NCC2CCCC2NC(=O)C(C2CC2)C2CC2)ncnc(O)c1F N1(C(C=Cc2c(C)ccs2)=O)CCC(CNC(C23CCCC2CCC3)=O)C1(C)C c1(CCS(N2CCC(NCCOCCOC)C2)(=O)=O)ccc(C#N)cc1 c1(C(=O)NC2CC(CC(=O)NCCCc3ccccn3)C2)cc(Cl)sc1Cl C(N=c1nc(N2CCC(C)(F)C2)c2ccc(C)cc2[nH]1)c1nc(C)[nH]n1 c1(OC)nc(Cl)ccc1C(=O)NC1CCCC(CN(C(=O)CNC=O)C)C1 C1(NC(c2nc(COC)oc2)=O)CC2(C1)CN(C(=O)CC1CC(F)C1)C2 c1(CC(=O)NCC(CC)NC(C2CCN2CC)=O)cccc(OC(F)(F)F)c1.C(C)CC C(=O)(C(C(F)(F)F)C(F)(F)F)N(C1CCN(C(CN(C)CC)=O)CC1C)C C1(N(C(C(=O)OC)=O)C(C)=O)CCCC1C(=O)OC N1(C(C2N(CCC)CCC2)=O)CCC(F)(CNC(c2nonc2C)=O)C1 N1(C(c2ncn(-c3cn(C)nc3)c2)=O)CCN(C(c2cnns2)=O)C(CF)C1 N1(C(CC)(CC)C(N)=O)CCC2(CC1)OCCO2 C1(NC(C2(c3ccccc3)CCC(=O)C2)=O)CN(C(C2(F)CC2)=O)CC2(CC2)C1 N1(CC(=O)N(C(C(=O)OC)C)C2CC2)CCC(F)(C(F)F)C1 C#Cc1cccc(C(=O)NC(CNC(=O)CC2(C(=O)OC)CC2)CC(F)(F)F)c1F C1(O)(OC)CC(C(=O)NC)C1.C(C)(C)(C1CN(C(C2(C(=O)N)CCC2)=O)C1)C1CC1 c1(C(N(CC(CN(C(C(C)CCN(C)C)=O)C)O)C)=O)cccc2ccsc12 CC(C)CCCC(C)NC(C1C=CCCN1C(c1cnc(Cl)s1)=O)=O c1(C(N2CC(NC(C(CC)F)=O)C(c3ccccc3F)C2)=O)cc(Cl)ccc1F c1(CNC(=O)CSC(F)(F)F)ccc2c(c1)CCN(C(C1C3CCC(=O)C13)=O)C2 c1(C(=O)NCC(c2ccc(OC)cc2)N)ccc2c(C)cc(Cl)nc2c1 C(CCC(=O)NCC1CC(C(=O)NC2CC2c2ccn(C)c2)C1)OC C1(CCNC(c2c(C)n(C3CCC3)nc2)=O)CC2CCC(C1)N2C(C1CCC1)=O C(N=c1[nH]c(=NCC(C)(CN(C)C)CO)[nH]c2c1COCC2)c1c(C)nn(C)c1 c1(C(N(C2CN(C(=O)C=CBr)CC2F)C)=O)cnn2ccn(C)c12 Cc1cccc(CCNC(C2(NC(=O)C=CCCC(C)C)CC(F)(F)C2)=O)n1 C1(C(=O)OC)CCC(C(N2CCC(CNC(=O)CC3CCCCC3)C2)=O)CC1 C(=O)(C1=NOC(CNC(=O)C(C)(C)C#N)C1)N(C)CC1(O)CCCCC1 CCCC(C)(CC)C(=O)NCC1C2CC1N(C(=O)C=Cc1csc(Br)c1)C2 c1(CN2CC(C(=O)NC3(C(=O)OC)CC3)C(O)CC2)cc(OC)c(Br)cc1C Cc1cc(-c2ccc(-c3nccn3CCC3CCC(C)(C)CC3)cc2)ccc1I C(=O)(CCC[N+](=O)[O-])NC(CCCC)CNC(C1CCCNC1=O)=O C1(C(=O)NCC2CCC(NC(CCN(CC)CC)=O)C2)CC1C1CCCCC1 N1(C(C2N(CC)C(=O)CC2)=O)CC2CN(C(c3cc(C#N)ccc3Cl)=O)CC2C1 CC12CC1CCN2C(c1cc(C2(C(=O)O)CC2)on1)=O c1(N(C(CS(CC)(=O)=O)=O)C2CNCC2F)nc(C)nc2ccccc12 c1(CN2C(CC#N)CN(C(c3cscn3)=O)CC2)c(F)c(F)c(F)c(F)c1F CC1CN(C(=O)C(C2(O)CN(C(C3C4(CC4)C34CC4)=O)C2)F)c2ccccc21 c1(C(=O)NC2C(CNC(=O)CCc3cocn3)C2)cc2c(nn1)CCC2 Cc1cc(C(N2CC3CC2CN3C(C2CCCC(C)C2)=O)=O)c(Cl)cn1 C1(CC(=O)N(C)CCC2(C)CCCO2)C2CN(C(=O)COCC3CCCC3)CC12 FC1(F)C(c2nc(-c3ccncn3)nn2C2CCSCC2)C12CCOCC2 C(=O)(CCCS(C)(=O)=O)N(C1CN(C(c2ccc(O)c(F)c2)=O)CCC1O)C C(=O)(C(F)C(F)(F)F)NC(C1CCCN(C(=O)Cc2cscn2)C1)C N1(C(CC(C=C)CC)=O)CCC2(CC(NC(C3CC4(C3)CC4(F)F)=O)C2)C1 C(CC(C(C)(C)C)NC(=O)Cc1cccs1)N(C(C(CC)C#N)=O)C c1(CCC)cnnc(C(=O)NC2CCC(CNC(C34CSCC3C4)=O)C2)c1 CCC(C)(C#N)C(=O)N1CCC(CC(=O)Nc2cnn(C3CC3)c2)CC1 Cc1cccc(Br)c1C1(NC(C2CCCC2C)=O)CC1 N1(C(c2cc(C)on2)=O)CC(C)OC2(CCN(C(c3cn(CCO)nn3)=O)C2)C1 C1(CC2(C(=O)OCC)CCCO2)CON(C(=O)c2cncc(C(F)(F)F)n2)C1 N(C(=NCCSC)NCCc1ccncn1)CC(COC)Oc1ccccc1 N1(C(C(CC=C)N(C(C)=O)CC)=O)CC2(C(N3CCCC(O)C3)=O)CCC1CC2 N1(C(C(CC)OC)=O)CCCC2(CCC2NC(C2CC(C(C)C)C2)=O)C1 c1(CC(=O)NCCC(C)NC(C2(C)CC2(Cl)Cl)=O)c[nH]c2cccnc12 CS(=O)(=O)c1cc(C(=O)NCCC2CCN(C(=O)C#CC3CCCO3)C2)co1 N(C(=Nc1ccccc1)NCC1CC(S(C)(=O)=O)C1)C1C(C2C(C)C2)C1 c1(C(N2CCC3(C(NC(=O)Cc4cn[nH]c4)C3)C2)=O)cc(F)cc(F)c1Br N1(CC(CCNC(=NC)NC2CN(C)CC2O)OC)C(=O)c2ccccc2C1=O n1(CC(=O)N(CCCNC(=O)CC2CCCOC2)CC)nc(C)cc1C c1(C(=O)NCC2N(C(CC(C)n3cccc3)=O)CCC2)ccc(S(C)(=O)=O)[nH]1 c1(C(=O)NCC(CC)N(C(=O)C(c2ccc(F)cc2)O)C)cc(C)n(CCO)n1 C1(C(=O)NC(C)C(CO)NC(C2CCN(C3CC3)CC2)=O)CC(C)(C)CN1C c1(OC)cccc(C(=O)NC2(CNC(C3CCCC3(F)F)=O)CC2)n1 c1(CC)ccc(N)c(C(=O)NC2CC2CNC(=O)C=CC2(C)CCOCC2)c1 N1(C(c2cc(COC)[nH]n2)=O)CCN(C)C(CNC(=O)CC2(C)OCCO2)C1 C=CC1(NC(c2conc2C(=O)OC)=O)CCCCC1.C12CC(C1)CNC2=O c1(C(N(CCCCN(C(COC(C)C)=O)C)C)=O)ccc(F)c2occc12 Cc1cc(Br)c(Br)cc1C(=O)Nc1cc(CO)ccn1 C1(NC(c2n(C)cnc2)=O)CN(c2cnc(Cl)cn2)CC2(CCC2)C1 C(=O)(CCCCCN(C)C)N1CCC(N(CC#C)C(C2CCC2CSC)=O)CC1 C1(OC)CCCCC1C(=O)NCCC(C)N(C)C(c1cccc(CC(C)C)c1)=O CN=c1[nH]cc(C(=O)OC(=O)CN2CCOC(Cn3cc(OC)cn3)C2)o1 N1(C(c2nc(OCC)oc2)=O)CC(C)CN(C(=O)CC#N)C(C)C1 CC1CN(C(=O)C=CC(=O)NC2CC2)CCCN1C(C12CCC1C2)=O c1(C(N(CCNC(C(CC=C)CC)=O)C2CCC2)=O)cc2ccc(CC)cc2[nH]1 c1(C(C)=O)c[nH]c(=NCc2noc(C3CC3)c2N(C)C(c2ccccc2)CCC)cc1Br c1(C(c2ccccc2)NC(=O)NCC2C3(CN(CCCC)C3)C2)cccc(Cl)c1 C12C3CC4C(C3NC1=O)C24.C(=O)(C1=C(Cl)CCC1)N1CC(=O)N(CCO)CC1 C=CCC(C(=O)NC(CNC(=O)Cc1ccc(O)c(F)c1)CO)C(C)C c1(OCC)ccccc1NC(=O)NCC(CCO)OC C1(NC(C(CC=C)NC(=O)CC2OCCO2)=O)CCCOC12CCC2 N(C(=NCCc1cccc(C(=O)N(C)C)c1)NCc1nnc(CO)s1)C(CC)C c1(C(C(=O)NC2CN(C(c3cnc(C)s3)=O)C2)O)cccc(F)c1 c1(OC)cc(C)ccc1C(N1CCCC1CNC(=O)C(c1ccc(F)cc1)F)=O C(=O)(CC1CCOc2ccccc21)NCC(C)NC(c1cc(=N)[nH]c(Cl)n1)=O c1(C(N(C2CCCCC2O)CCC)=O)cc2c(-c3nn[nH]n3)cccc2[nH]1 CCCCC(F)C(=O)NCC1CN(C(C2CN(C(C)C)C2)=O)CCCO1 C1(NC(CN(C2CCCC2)C)=O)CCCC(NC(c2cc(Br)nn2C)=O)C1 N1(C(C2C=CCN(C(CCN(CCC)C)=O)C2)=O)CCc2ncsc2C1 Cc1ccc2nonc2c1C(=O)N(CCCCNC(=O)CCCCCO)C CC1CN(C(C2CCCC2CNC(c2cncnc2)=O)=O)C(C)C(C)(C)O1 N1(C(c2cc(C)sc2)=O)CC(NC(=O)C(C)Cn2cccn2)CC(F)C1 c1(CNC23C(NC(=O)OC(C)(C)C)(CCC2)C3)cc2c(nc1O)CCCC2 C(C(C)(C)CC(=O)N(C)CC1COC(=O)N1)NC(C(C)c1cccs1)=O C1(C(=O)NCCC(=C)CNC(=O)CCNC(=O)NC)CCCC12CCOCC2 c1(OC)c(C(N2CCN(C3CC3)C(C)C2)C(=O)NC2(C)CC2)cccc1O c1(C(=O)NC2C(CNC(C(C)CF)=O)CCCC2)cn2cc[nH]c(=O)c2n1 c1(N(S(C)(=O)=O)C(c2scc(-c3c(COC)cccc3)c2)=O)cccc(C)c1Br CC(C)C(CCNC(=O)C(c1ccoc1)NC(=O)C(C1CC1)C1CC1)N(C)C c1(C(=O)NC2C(C)CN(C(CCC#C)=O)CC2C)ccc(S(=O)(=O)CC)cc1 CC(C)CC(CNC(c1ccc(C(N)=O)o1)=O)C(=O)N(C1CCN(C2CC2)C1)C C(CC(=O)NCc1occc1C)(C1CC1)NC(C1CN(C(=O)NC)C1)=O C1(C(=O)NCCN(C(COCC=C)=O)CCOC)CCc2ccccc2C1 C1(N(C(Cc2ccn(C(C)C)n2)=O)C)CCCN(C(=O)C(C)C2CCC2)C1 N1(C(C2(CC=C)CCOCC2)=O)CC2CC(NC(=O)Cc3cn[nH]c3)C1C2 c1(C(=O)OC)nc(NC(c2conc2C(C)C)=O)sc1Cl.C12CC(C1)NC2=O c1(C(=O)NCC(C)(C)NC(c2cccc(C(N(C)C)=O)c2)=O)coc2c1CSC2 c1(C(N(C2CCS(=O)(=O)C(C)C2)CC)=O)cc2c(OC)ccc(C)c2[nH]1 c1(CC(=O)NCC2C=CC(NC(C3(CC)CCOC3)=O)C2)n[nH]c2ccccc12 N1(C(CCCCCOC)C(=O)NCCC2(C)CC2)CC23CCCCC2(COC3)C1 c1(CC)noc(C(C)NC(=O)COC2CCOC2)n1 N(C(=NCCc1ccccc1)NCC(c1ccc(Cl)nc1)(C)C)CC(C=C)(C)C C(=O)(C(CC)CCCCC)NC(CC#CC)C(=O)NC1CN2CCCC1C2 c1(OCC(=O)NC2CCCCC2CNC(c2nsnc2O)=O)ccc(Cl)nc1 N#Cc1nccnc1N1CCC(CNC(c2ccc(-n3ccnc3)nc2)=O)CC1 C(=O)(C1=C(C#N)CCC1)NCCC1N(C(C2C(CC)C2)=O)CCSC1 C(=O)(C1COc2ccc(F)cc21)N1CCN(C(=O)CCc2cc[nH]n2)CC1CO CCCC(CC)CCC(=O)NC1CC12CC(NC(=O)C1=C(Cl)CCOC1)C2 c1(CC)oc(C(=O)NCC2C(C)CCN2C(=O)CCc2cncn2C)cc1C S(=O)(=O)(c1ccccc1C(=O)NC1CC1C(=O)Nc1ccc(I)cc1Cl)N(C)C C1(NC(C2(C=C)CCC2)=O)CC(OC)CN(C(c2nccn2CC)=O)C1 c1(CCCNC(c2cscc2-c2nn[nH]n2)=O)ccccc1Br N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(C2CCN(C(C3(O)CCSC3)=O)C2)CC1 C(C(C)(C)C1=CCOCC1)Nc1cccc(C)c1C.N1(CCO)CC1 c1(COC2CCN(C(=O)COC3COC3)C2)cccc(Cl)c1 c1(OCCOC)ccc(C(N2CC(C(C)NC(C3CCCC3C)=O)C2)=O)cc1 C1(C2CC2)(CNC(Cc2c(C)ccs2)=O)CCN(C(=O)C(O)CN(C)C)C1 c1(OCCN(C)C)cccc(C(N2CCCC2(C)CNC(c2cnsn2)=O)=O)c1 C1(C(N2CCCC(OCCC)C2)=O)CC2CCC(C1)N2C(c1cscc1C)=O CON1CCC(CC(=O)NC(C)CCCNC(=O)CC23CC(C2)C3)CC1 n1(CCCC(=O)NC2CCC(CNC(CC3(C)CC3(F)Cl)=O)C2)ccccc1=O n1(CC)ccc(C(N2CCC2CNC(C2(CN(C)C)CCCC2)=O)=O)n1 c1(C(=O)NC2CN(C(C3(OCC)CCOC3)=O)C(C)(C)C2)cc(F)c(C)cc1O c1(COC)cc(C(=O)NCC(C(=O)N2CCC2C2CCOCC2)N(C)C)n[nH]1 C1(CNC(c2c(C)n[nH]c2C)=O)CN(C(=O)CC2COC(C)(C)C2)CC1(F)F C1(C(=O)NCC(=O)Nc2cn[nH]c2)CC(F)(CNC(CCC)=O)C1 C12(NC(CC3CCC(NC(C)=O)CC3)=O)CCN(C(=O)C3=COCCC3)CC1C2 c1(C(C)SCC)ccc(S(=O)(=O)N(CCNC(=S)NCCOC)C2CC2)o1 c1(N2CCC(C(C)(C)C)CC2)nccc(=NC(CCO)c2ccccn2)[nH]1 c1(COC)cc(C(=O)NCC2(NC(=O)CCc3cnoc3)CCCC2)cs1 C(=O)(C1=CCN(C(c2ccn(COC)n2)=O)CC1)NC(C#C)C1CCC1 C1(CCCC)CCC(C(N2CC(NC(c3cn(C4CC4)nn3)=O)C2)=O)CC1 C#CCCC(O)C(=O)NC1C2CC1N(C(=O)C=Cc1ccc(C)cc1)C2C Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)N1CC2CN(C(=O)CO)C2C1 c1(C(N2CC3CCC2CN3C(=O)C2=NOCC2)=O)c[nH]c2c(Cl)cccc2c1=O Cc1nn(C(C)C)cc1C(N1CCC(N(C(=O)CCc2ccoc2)C)C1)=O C=CC1CCCN(C(=O)C(C)(C)CNC(C2CC3CC2CC3O)=O)C1 c1(C(CNC(C=C(C)CNC(=O)Cc2ccn(C)n2)=O)O)cn(C)cn1 c1(CN(CC)Cc2cccc(C(F)(F)F)c2)c(Br)nc2n1CCOC2 C1(OC)(CNC(=O)CC2COCCOC2)CCN(C(C2(O)CC2)=O)C1 c1(C(=O)NCCN(CCC)C(c2cc3scnc3[nH]2)=O)ccc2cncn2c1C C(=O)(CC1=Cc2ccccc2C1)N1CCCC(NC(C=CC=CC)=O)C1C C#CCCC(O)C(=O)N(C1CN(C(=O)Cc2cc(Br)cs2)C1)C C#Cc1cnn(C)c1C(N1CCC(N2CCC(NC(C3(C)CCC3)=O)CC2)C1)=O N1(C(C(c2ccc(Cl)cc2)=O)=O)CC2CCC1C(NC(N1CCCCCC1)=O)C2 c1(CC(=O)N(C(CNC(c2coc(O)n2)=O)C2CC2)C)cc(F)cc(F)c1 c1(C(CC)N(C(C)CCBr)C)ccccc1F c1(C(=O)NCCC(C)N(C(C(C)c2cncs2)=O)C)cc2cccc(F)c2o1 C(=O)(CC1CNc2ccccc21)NC1CCN(C(c2c(C)c[nH]n2)=O)CC1 C1(C)(NC(CN2CCC(C)(C)C2)=O)CCC(NC(c2ccsc2)=O)CC1 C1(CC(=O)NC(C#C)(CC)CC)CN(C(c2ccc(C(C)C)o2)=O)CCC1C C(C(C)(C)CC=C)NC(c1n(CC=C)nnn1)c1cnn(CC(F)(F)F)c1 C#CC1CCCCN1C(C1(C)C=CCN1C(C1CCC1C(C)(C)C)=O)=O c1(CC)c(C(N2CC(CNC(=O)CSc3nncn3C)C(C)C2)=O)nnn1CC CC1(CC(N2CC(NC(C3CSCCS3)=O)C2)=O)CCOC1 c1(C(=O)NCCCCCN(C(CC=CC=C)=O)C)nc2cc(F)ccc2s1 c1(C(N2CCCC(O)(CNC(C(CC)(C)C#N)=O)C2)=O)cc2cc[nH]c(=O)c2s1 C1(NC(c2c(CC)noc2)=O)CCCCC1NC(c1cnn(CC(C)C)c1C)=O CCCCC(C)CCC(=O)N1CC(NC(C2CCCS2)=O)C(F)C1 c1(NC)ccc(OC)cc1C(F)(F)F.C123CCCC1(C2)CNC(=O)N3 C(=O)(C(O)CSC)N1CC(CC(=O)N(C2(C(=O)OC)CC2)C)C1 n1(C(C)C)[nH]c(CC(=O)NCC(C)(C2CC2)NC(=O)CC2COC(=O)C2)cc1=O O=C(CS(=O)C(F)(F)F)NCCC1CSCCN1C(c1cc(Cl)cs1)=O c1(OC)ccc(C(N2CCC(CCNC(=O)CNS(C)(=O)=O)CC2)=O)c(OC)n1 C1(C(N2CCC(N(C(=O)CC=CC(C)(C)C)C)C2)=O)C2CNC(=O)C12 C(CC(CC)C(=O)NC(C)(C)CCC(=O)NC1CN(CC)CC1C)=CC c1(C(N(CC(C)NC(C2OCCC2C)=O)CC)=O)ccnc(OCC(F)(F)F)c1 Cc1nn(CC(=O)NCC(C)(CO)NC(=O)Cc2cnc[nH]2)cc1Cl c1(OCC(=O)NC(CC(C)NC(C2CC(CC)C2)=O)C)ccc(C)cc1F CC(=O)C(C)CC(C)C(=O)N1CC(O)CC1CC(=O)NCCC(C)C(=O)OC C(=O)(C1=CCCC1)NCC1CCN(C(C2(O)CCSCC2)=O)C1 CC1(CNC(=O)COC2CCCCC2)CCC(NC(=O)COC(F)F)CC1 c1(OC)cc(C(=O)NC2CCCC(CNC(c3cccc(F)c3)=O)C2)cc(C)n1 Cc1cc(C(=O)NCCN(C(=O)C(C)CC#N)C(C)C)cnn1 Cc1ccc(C(N2CCN(S(=O)(=O)CC(=O)ON)C3CC23)C(=O)NC(C)C)cc1F CCC(C)(C)CC(=O)N(CCCNC(=O)CCCc1cc(O)ccc1C)CCO C(=O)(CCCCCC(C)(C)C)NCCC1(O)CN(C(CCC2CCC(C)O2)=O)C1 c1(C(N2CCC(C)(NC(c3ccn(C)n3)=O)C2)=O)ccc2c(c1)CCC=C2 C1(NC(C(c2c(C)noc2C)CC)=O)CC2(NC(C3(CCO)CC3)=O)COC1C2 O=C(C1=CCOCC1)NCCC1(C(N2CC(O)(C(F)(F)F)C2)=O)CC1 C#CC1CCCN(C(=O)CC2CN(C(=O)Cc3cnnn3C)CC23CC3)CC1 c1(C(N(C2CCN(C(C3C(OCC)C3C)=O)C2)C)=O)cc2nn[nH]c2cc1F CCCC(C)(C)C(=O)NC1CN(c2nnn(C)n2)C1 N1(C(C2CCCC(C)(C)O2)=O)CC(C2CCCCN(C(=O)COCC(F)F)C2)C1 O(NC(=O)C(CCF)NC(C1CC2CCC1CC2)=O)C(c1ccccn1)C CC(C)C(C(=O)N1CCCCC(CNC(=O)C(F)(F)CO)CC1)C(C)C C1(c2cn(CCNC(=O)CC3CCCC3)nn2)CCN(C(=O)COC)C(C)C1 CC(C)(CCS(C)(=O)=O)NC(c1cc(C(N)=O)cs1)=O C12(C(C(=O)NC3CCC3NC(=O)CC(=O)N(C)C)OC)CCC(CC1)C2 CCCCC(O)C(C)C(=O)N1CCC(NC(=O)C=CC2CCC2)C(F)C1 c1(C(=O)NC2C3CCN(C(C(CN(C)C)O)=O)CC32)ccc2nncn2c1 CC(O)C(F)(F)C(=O)NCc1cccc(C(=O)NC2CCC3CC23)n1 c1(C(N2CC3(CCN(C(C(=O)N(C)C)=O)CC3)C2)=O)cccc2c(Cl)ccnc12 c1(C(N2CCC(CNC(C3CC3C(F)(F)F)=O)C2)=O)ccncc1Br c1(C(N2CCC(O)(CN(C(CCCOCC)=O)C)C2)=O)cc(Cl)ncc1F C(=O)(C(F)(F)C(C)(C)O)N1CC(C(N(CCCC)OC)=O)C(C)(C)C1 CC(C)(CCNC(=O)C1=C(Cl)CCC1)C(=O)NCc1cccc(C#N)c1 CC(C)CCCC(C)NC(=O)OCC1CCN(Cc2ccccc2)C1 C1(NC(C2(C3N(C(CCC=C)=O)CCC3)CC2)=O)CCC(C)CC1 c1(C(N2CCC(NC(c3c(Cl)cn(C)n3)=O)C2)=O)cc([N+](=O)[O-])cn1C C1(c2onc(C(C)(C)OC)n2)(NCc2nc(Cl)c(Cl)s2)CCSCC1 C1(C2CCC(c3c(C)ncs3)O2)CCN(c2nnc(-c3cncn3C)o2)CC1F CC(CNC(=O)C(c1ccccc1)O)C(=O)N(C1CCC1(C)C)C C(C(COC)CC(=O)N(C(C)CCNC(c1cccc(=S)n1O)=O)C)OC C1(CNC(CCOCCC)=O)CCC(C)N(C(=O)CSc2cn[nH]c2)C1 CCC(C(=O)N1CCC2CC12C(=O)NCCCN(C)C)C(F)(F)F C1(OC)(CNC(C2CC(C)=NO2)=O)CCN(C(c2ncccc2F)=O)CC1 c1(OC)cccc(N2CC(C(=O)NCC(C)(C)NC(=O)C(=O)N(C)C)CC2=O)c1 N1(C(C=CC)=O)CCC(C)C(CNC(c2cnn(C)c2-c2ccc(F)cc2)=O)C1 Cc1cn2cc(C(N3CC(NC(c4cc[nH]n4)=O)CC(F)C3)=O)sc2n1 N1(C(C2CC(=O)NCC2)=O)CC2(C(=O)NC(CO)(CO)CO)CCC1CC2 CC(C(=O)N1CC2CC1C2C(=O)NCc1ccc(Cl)cn1)S(N)(=O)=O C1(Cl)(C(=O)NCCCN(C(C(C)SCC)=O)C2CC2)CC12CCC2 C(=O)(CCC(C)(C)C)NC(CCCC)CNC(c1ccc(F)nc1)=O C1(C(=O)NC2CC(CCNC(c3c(CCC)nsc3N)=O)C2)CCOCC1(C)C N1(C(CC2N(C)CC=CC2)=O)CCC(NC(=O)CCc2nc[nH]n2)C(CO)C1 C1(NC(CCNC(=O)OC)=O)CC(O)CN(C(=O)CSc2nnc(S)s2)C1 C1(C(=O)NC(CNC(c2c(C(C)(C)C)n[nH]c2)=O)C2CCC2)CCCCN1N=O c1(CC(=O)NCCN(C(COC(CC)(C)C)=O)CCOC)ccc(O)nc1 c1(CC(=O)NCCOCCN(C(c2cc(C)ncc2)=O)C)ccc(F)c(C)c1 C(=O)(C(C(C)C)NS(N)(=O)=O)NC(C(C)C)CNC(c1cnc(S)[nH]1)=O CC1(C)CC(Nc2ncc(C(F)(F)F)cc2Cl)CN1C(=O)Cn1cncn1 O=NN1CCCCC1C(N1CCOC(CCNC(c2ccc(O)cc2F)=O)C1)=O N1(C(=O)OC(C)(C)C)CC(NCC23CCCC2(CO)C3)CC2(CCC2)C1 C1(OCC)CC2(C1)CC2NC(=O)C(O)CNC(=O)COc1ccccc1 c1(C(N2C(C)CN(C(C3CCC4CC34)=O)CCC2)=O)ccc(F)c2ccncc12 CCC(C)CCC(=O)N1CCCCC1C(C)(C)CNC(c1cccc(O)c1F)=O N1(c2nc(C(=O)OC(C)(C)C)n3c2cccc3)CCn2ncc([N+](=O)[O-])c2C1 C1(CCC(=O)NCCCCN(C(=O)C(C)C2CCC2)CCOC)CCCCO1 N1(C(C2CCC(C(C)C)NC2=O)=O)CC(C)(C)C(NC(=O)C2=CCC2)C(C)(C)C1 CC(C)CC(C)(CN=c1ccnc[nH]1)NC(c1cnc(C(C)(C)C)[nH]1)=O CC1Oc2cc(-c3nnc(-c4nccn4C)o3)ccc2NC1=O n1(CCC(N2CCN(C(CC(=O)NC)=O)C(CO)C2)=O)cnc2ccccc12 N1(C(C2CN(C(C3(C)CC(=C)C3)=O)CC23CC3)=O)CCCN(C)CCC1 c1(C(=O)NCC(C(C)C)NC(CCC(C)=O)=O)ccc2cnc(C)cc2c1 c1(C(CNC(C2CC=CCO2)=O)NC(CSCC#C)=O)ccc(F)cc1F N1(Cc2cnc(C)[nH]2)CC2(CC2)CC1C(=O)Nc1ccc(C(F)(F)F)cc1C CCC(F)(F)C(C)(C)C(=O)N(CCC(C)NC(C1(C2CCCO2)CCC1)=O)C C(CC(C)(C)C(=O)N(CCC(=O)NCC1(O)CCCC1C)C)SC c1(C(=O)NCCCCCN(C)C(C2CCC2F)=O)cn(CC(F)(F)F)cn1 C#CCCCC(C)C(=O)N1CCCC(NC(c2ccoc2C(C)C)=O)C1 C1(C(=O)NC2CCC2C(=O)NC(C2CCCCC2)CO)CC2(CCC2)CO1 Cc1ccccc1CC(C)C(N1CC(NC(=O)C(C)(C)CN(C)C)CC1CO)=O C=C(C)C(CC(=O)NCC1CC(NC(=O)C(C)Sc2ccc(C)cc2)C1)OCC N1(C(c2c(C)sc(O)n2)=O)CCCCC(NC(C2(CC(C)C)CCCC2)=O)C1 N1(C(c2c(CC)n[nH]c2)=O)CC2(CCCC2NC(c2csnc2C)=O)C1 N1(C(COCCC)=O)CCCCCC(NC(c2ccnc(-c3ncc[nH]3)c2)=O)C1 N1(C(c2c(C)[nH]cc2)=O)CC(C)CCC1CNC(=O)CCc1cnoc1 CC(CCO)N=c1[nH]c(N2CCC(CF)C2)nc2ncn(C)c12 C1(C(N(CC(=O)NCC2CC3(CC3)CO2)C)=O)CC(C)(C)CO1 C1(CC(=O)NC(C(C)(C)OC)C)CCN(C(=O)CC2(C)CC2)CC1 C(CNC(C1CCC=CCC1)=O)(CC(=O)NC(C(O)CO)C1CC1)OC N1(C(=O)CCc2ccc[nH]2)CCOC2CN(Cc3ccc(OC(F)F)nc3)CC12 C#CC1CN(C(c2c(Br)ncn2C)C(=O)Nc2ccc(C)cc2)CC1O Cc1cccnc1C=CC(N1CCC(NC(=O)CCc2cscn2)CC1C)=O C(=O)(C1=NN(C)C(=O)CC1)N(CCCNC(C(c1cnccn1)C)=O)CCO C=CCCCCC(=O)N1CC2CC1CN2C(c1cc(CC)[nH]n1)=O c1(-c2cn(CC(CC(=O)NCCOCC)O)nn2)cccc(C2(O)COC2)c1 C#CCCCCCCCC(=O)N1CC(O)(C(C)NC(=O)C(C)CC)C1 Cc1cccnc1CC(=O)N(C1CN(C(c2c(CO)noc2C)=O)CC1F)C S(=O)(=O)(c1c(C)cccc1Cl)N1CC(COC)N(Cc2csc(Br)c2)CC1 n1(CCOC)cc(C(=O)NCC2C=CCN2C(=O)COCCOC)c(C)n1 c1(C(=O)NC(C)CCN(C(=O)C(C)n2cncn2)C)cccc(CO)n1 n1(CC)c(C)nn(CC(N2CCC(CCOC)(NC(=O)C3=COCC3)C2)=O)c1=O CC(C)(CC(F)F)C(=O)NCCCCN1CCCN(C(C2CC(O)C2)=O)CC1 C(=O)(C1=CCCSC1)N1CC(C(C)NC)C1.C=CC1(C(=O)NC(C)=O)CCC1 C12(C(=O)OC)CCC(C(=O)Nc3ccnn3CSC3CCCCO3)(CC1)C2 C12(C(N(CCNC(C(C)(C)SC)=O)C3CC3)=O)CCC(CC1)C2 Cc1ncnc(O)c1C(=O)NC1CC2CC(NC(C3(C(F)(F)F)CC3)=O)C2C1 Cc1cccc(F)c1CC(=O)NC1CCN(C(=O)Cc2cnn(C)c2)CC1CO Cn1cc(C(=O)NC2(C)CN(C(=O)Cc3ccnc(C(F)(F)F)c3)C2)n(C)c1=O CC(CN(C)C)CCC(=O)NCCC1CC(NC(c2ccc(C(F)F)o2)=O)C1 C1(NC(C2(C)CC2(F)F)=O)CCC2(CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2)C1 N1(C(=O)C(F)Cc2ccccc2)CCN(C(c2cnc(Cl)s2)=O)C(CC2CC2)C1 c1(C(=O)NC2(CC(=O)NC(C3(CO)CC3)C)CCC2)ccc(=O)n(C)c1 CC(C)CC(O)CC(=O)NCCOc1ccn(C)n1 C(C)(C)(CCCCC(=O)N1CCN(C(=O)CC2=CCCC2)C(C)C1C)OC C1(NC(CCC(C)(C)NC(=O)C2=CCCCC2)=O)CCCCCCC1O C1(C(N(CCC(C)NC(CCOCC)=O)C)=O)Cc2cc(C)ccc2S1 c1(C(N2CC(O)(CNC(c3cccc(C)c3F)=O)C2)=O)cnc2c(F)cccn12 CCC(C(=O)NC1CC(CNC(c2cnc(C(F)(F)F)nc2)=O)C1)C(C)O C1(CC(=O)NCC(C)(C)CCNC(=O)C=Cc2ccccc2)CC(=O)NC(=O)C1 N1(C(c2c(C)c(-c3ccccc3)[nH]n2)=O)CCN(S(C)(=O)=O)C(CC(=O)O)C1 C1(NC(c2ccnc(CC(C)C)n2)=O)CC2CC1N(C(=O)C(F)F)C2 N1(C(C2(N(C)C)CCC2)=O)CC2CC(C1)N(C(c1nnn3c1CSCC3)=O)C2 c1(C(=O)NCCNC(c2occc2-c2ccccc2)=O)ccnc2[nH]nnc12 Cc1cc(CC(=O)NCC2(C(C3CC3C)=O)CC2)sn1.C1(=O)CCSCCN1 c1(CCNC(c2n(CC=C)nnn2)(C)CCSC)ccc(C)nc1 N1(C(COCCC#C)=O)CCC(CNC(c2cc(F)ccc2C)=O)C(O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC2(CCN(C(c3c[nH]c(=S)cn3)=O)CC2)C1 C(CCCCCC(=O)N(C1CCN(C(c2c[nH]c(=N)nc2C)=O)CC1C)C)SC N1(C(COc2ccc(C)cc2F)=O)CCCC12CCCN(C(=O)C(O)C1CC1)C2 N1(C(CCC#C)=O)CC2CN(C(c3sc(C(=O)OC)cc3N)=O)CC2C1 c1(NCC(c2nnnn2Cc2ccco2)NC(N)=O)ccc2cnccc2c1 c1(C(=O)NC(C(C)C)CNC(=O)CC2COCCN2C)ccc(N)c(SC)c1 c1(C(=O)NCC23C(CN(C(c4c(C)nsc4)=O)C2)C3)ccc2nnc(O)n2c1 c1(C(=O)NCCN(C(=O)CN2CCC(O)CC2)CC)nc(=N)cc[nH]1 C(C)(CN=c1ccn(CCc2nc(C)cs2)[nH]1)(c1n(CC(=C)C)nnn1)OC CCCCCCC(C)NC(c1c(Cl)ccnc1Cl)c1nnnn1C1CC(F)(F)C1 C#CCC(CC(=O)NCCCCC1CC1C)NC(=O)CCCC(=C)C C1(CC(=O)NC(c2ccccc2)CO)CCN(C(C2CC3CC3C2)=O)CC1 C(=O)(C1Cc2ccccc21)NC(CN(C(C(C=CC)O)=O)C)(C)C Cn1cc(C(N2CC(CCCCNC(=O)C=Cc3cocn3)C2)=O)c(C(F)(F)F)n1 N1(C(C2N(C(CC3(C(=C)F)CCC3)=O)CC=CC2)=O)CC2(C1)CC(C)(C)C2 c1(C(N2CC(CCNC(COCC=C)=O)OC(C)C2)=O)ccc2nc(S)oc2c1 n1(C(C)C)cnc(CNC(c2coc(CNC(=O)C(C3CCCCC3)C)c2)=O)n1 NS(=O)(=O)CCCCN.c1(C(C2C3COCC23)CCC2CCCO2)nnn[nH]1 c1(OC)ccc(C=CC(=O)NCCC(C)NC(c2ccc(F)c(F)c2)=O)cc1 c1(CCC)c(C(=O)NCCOC2CCN(C(=O)CC3CC3C)CC2)nnn1CC C(=O)(C(O)CC(F)(F)F)NCC1CN(C(=O)NC2CC(O)(C(F)F)C2)C1 N1(C(=O)C=CC2CCOCC2)CC2CC1C2C(N1CC(CC2CC2)C1)=O C(=O)(C1=Cc2ccccc2OC=C1)N1CC(OCC)C(CNC(=O)CCF)C1 N1(C(c2c(C)nccn2)=O)CCOC2(CCCN(C(=O)COC3CC=CC3)C2)C1 Cc1ccc(F)c(CNCC23CCC(NC(=O)C(F)C4CCC4)(CO2)C3)c1 c1(C(=O)OC)ccc(C(F)F)cc1.N12CCC1C(=O)OCC2 C12(C(=O)NCC(C(C)C)NC(c3coc(-c4cccnc4)n3)=O)CCCC1C2(F)F c1(CCC(=O)NCC2CCC2NC(C2CC2c2nc[nH]n2)=O)ccc2ncsc2c1 C#CCC(C(=O)NC1(C(C)C)CC1)NC(=O)C=Cc1ccccc1 CC1OC2(C(=O)NCCN(C(=O)C3=CCOCC3)CCOCCO)CCC1CC2 c1(CN(C)CC2CN(C(C3CC(F)C3)=O)C2)cc2ccccc2nc1Cl C(C)(CCCCCO)NC(C1(C)CN(C(c2c(CCC)nco2)=O)C1)=O c1(C(=O)NCCC2(NC(c3cc(C)oc3C)=O)CC2)cc(Cl)ccc1C(N)=O c1(OCC)cc(CNCC(C)C(F)(F)F)c(C)cc1C Cn1nnc(C(=O)NCCC2CC(NC(=O)COCc3ccc(Cl)nc3)C2)c1N C(c1ccc2c(c1)CCO2)=CC(=O)NCC(CN(C(c1ncc(C)cn1)=O)C)C c1(C(=O)NC2C(NC(C(C)NC(N)=O)=O)C2)ncnn1C1CCOCC1 c1(C(=O)NC2C=CC(C(=O)Nc3ccc(C)cn3)C2)cc(F)cnc1Cl N1(C(C(c2cn(C)nc2)=O)=O)CCN(C(=O)COC2CC=CC2)C(C2CC2)C1 O=C(C1=Cc2cc(F)ccc2OC1)NC1CC(NC(C2CCC(O)C2)=O)C(O)C1 n1(CC(=O)NC2CC(NC(CC(C)(C)O)=O)C(O)C2)cnc2c1CCCC2 c1(COC)cncc(C(=O)NC2CC(CNC(c3cc(Cl)cnn3)=O)C2)c1 C12(C(=O)NCC3C(NC(=O)Cc4cc[nH]n4)CCC3)CCC(CO)(CC1)CC2 N1(C(CCCCNC(C2=NOC(C)C2)=O)=O)CCC2(CCOC2=O)C1 Cc1cc(C)c(C(=O)NCC(C)CNC(c2nc(C)sc2C)=O)c(C)c1 Cn1cc(C(F)(F)F)nc1C1CCCN(c2cc[nH]c(=N)n2)C1 C1(CC=C)(NC(=O)CCNC(c2ccsn2)=O)CCN(C(=O)C=C(C)C)C1 c1(SC)cc(Br)ccc1C(=O)CSc1cncnc1 Cc1ccc(C=CC(N2C3CN(C(c4ncoc4C)=O)CC23)=O)s1 N1(C(C(c2cnn(C)c2)C)=O)CC2CCC(C(N3CCOCC34CC4)=O)(C2)C1 c1(C(=O)NCCN(C(=O)Cc2cnnn2C)CC)ccc2nc(O)[nH]c2c1 C1(CNC(c2c(OC(C)C)cccc2)=O)CC2(C1)CN(C(C1CS(=O)(=O)C1)=O)C2 c1(CN(C(C)(CCl)C2CCCC2)CC2CC2)ccccc1 N1(C(COCCC)=O)CC2CCCN(C(c3cnn(C(C)C)c3)=O)C2C1 CC12CC(C(=O)NC3CC3CNC(c3nc(C4CC4)cs3)=O)(CCO1)C2 c1(C(=O)Nc2n(CC)ncc2)cc2c(-c3cc([N+](=O)[O-])ccc3F)cccc2s1 c1(C(=O)NCC2CN(C(C3(C)CCN(C)CC3)=O)C2)ccc2ocnc2c1 O=C(N=c1[nH]oc2cccnc12)C1CCCN(Cc2ccc(F)c(C(F)F)c2)C1 c1(C(N(C(C)CNC(=O)Cc2nc(C)sc2C)CC)=O)csc(=NC)[nH]1 N1(C(C(C#N)=CC2CC2)=O)CCCCC2(CCN(C(c3cnns3)=O)C2)C1 c1(CCC(N2CC(N(C)C(C34CCC3C4)=O)C(O)C2)=O)ccc(Br)cc1F c1(C(=O)NCC2(NCC)CC2)cccc2cnsc12.C1(C(=O)OCC)CC1CCC c1(C(=O)NCCCN(C(c2n(C)ncc2)=O)Cc2ccccc2)cc(N)ccn1 c1(C(=O)NCC)oc2ccccc2c1C(C)NCc1cc(OC(C)C)ccc1F c1(C(N(CCNC(CCC(=C)Cl)=O)C2CC2)=O)cc(S(=O)(=O)N(C)C)cn1C C1(C)(CC(c2n(-c3ccc(OC)cc3)nnn2)NCc2ccsc2)CCCCCC1 c1(NC(C2N(Cc3c(C)nn(C)c3C)CC2)=O)ccc(S(=O)(=O)C2CC2)cc1 C(C(C)(C)CC(C)NC(c1sc(SC)nc1C)=O)OC.C(C(=O)NC)NC(C)C N1(C(CN(CC)CC)=O)CC2(CCN(C(C3CC4C=CC3C43CC3)=O)C2)C1 N1(CC(=O)NCC2(CNC(C(C)(C)c3cccnc3)=O)CCC2)CCCS1(=O)=O N1(C(=O)C=CCN2CCCC2)CC2C(CNC(=O)CNC3CCCOC3)C2C1 N1(C(CNC(CCC(C)C)=O)=O)CC2CCCC2(NC(C23CC(C)(C2)OC3C)=O)C1 CC1(C)CC(NC(=O)COCC2CCOCC2)CN(C(c2cncc(N)n2)=O)C1 CCCC(CNC(=O)C(C1CCN(C(C2(n3cccn3)CC2)=O)C1)C)CCC c1(OC)nccc(CNC(C2CCC2CNC(=O)CC2(O)CCOC2)=O)n1 N1(C(C2CC(C)(C)OCC2)=O)C(C(=O)NOCCC(F)F)CC2CCCCC12 C1(NC2C(NC(C3N(C(=O)NC(C)C)CCC3)=O)C2)CCCC12OCCO2 CC1(C)CCCC(CC(=O)NCC23CC2CN(C(c2cccc(Cl)c2Cl)=O)C3)C1 C(CCCCCNC(c1cn(C2CCC2)nn1)=O)N(C(CCN(CCC)C)=O)C C(C(CC1CC1)C(=O)NCC(=O)OC(C)C)NC(CSCCOC)=O c1(C(=O)NCC2CN(C(C(C)SC)=O)CC2c2cncn2C)cccc(Cl)c1C C1(CNC(C(C(C)C)C)=O)CN(C(=O)CCN(C)C(=O)OC(C)(C)C)C(C)(C)C1 C(=O)(C(C)(C)C(=O)NCC(C)(C)C(=O)NCCC(F)(F)CO)N(C)C c1(SCc2n(CC)cnc2)cccc(S(C)(=O)=O)c1.c1(C)nc(CN)no1 c1(C(N(C(C)C(=O)NC23CC=CC(C2)OC3)C2CC2)=O)ccc2ccoc2c1 C1(NC(c2cc(C(F)F)[nH]n2)=O)CC2(C1)CN(C(c1coc(Br)n1)=O)C2 C1(C(N(C)CC2(NC(c3cn(CCC(C)C)nn3)=O)CC2)=O)CC2CC1CO2 C12(NC(CN(CCC)C)=O)CCCN(C(c3ccc(Cl)nc3O)=O)CC1C2 CCCC(CC)C(=O)NC1CN(C(c2sccc2F)=O)C(C)(C)C1 N1(C(CC=CC=C(C)C)=O)CC(C(=O)Nn2ccnn2)C(C)(C)C1 C#CCC(C(=O)O)NC(C1CC1(F)F)=O Cc1sc(N)c(C(N2CC3CCC3(CCNC(=O)C3=COCCO3)C2)=O)c1C N1(C(C(CC)C#N)=O)CCC(N=[N+]=[N-])(C(=O)Nc2cccc(C)c2C)C1 C1(NC(c2cn(C)nc2Cl)=O)CC2(C1)CN(C(C1CCCC1(F)F)=O)C2 N1(C(C(C(C)(C)O)F)=O)C(C(=O)NC2COC(C(F)F)C2)C2CC(O)C1C2 c1(CC)nn(C)c(CC)c1CC(=O)OCC.C12(CCOC3(CC3)C1)C(=O)O2 CCCCC(C)(F)C(=O)N1CCC(CNC(c2coc(C(F)F)n2)=O)(OC)C1 CC1CCC(NC(=O)CN(C)C2CC2)CN1C(=O)CCc1ccccc1O c1(C(=O)NCc2cccc(Cl)c2)n[nH]c2ccc(-c3ccnn3C3COC3)cc12 c1(CCC(=O)NCC2N(C(CCN(CCC)C)=O)CCCC2)ccc(Cl)c(Cl)c1 c1(NS(C)(=O)=O)cccc(NCC2C=CCCC2C(F)(F)F)c1 Cc1nc(C)n(CC(=O)NCCNC(c2cc(C(=O)C3CC3)cn2C)=O)n1 c1(CC2(CC)C(OCC)CC2NC(c2ccco2)=O)ccc(S(=O)(=O)CC#N)cc1 C1(C(=O)NCC(C)Cn2cccn2)CN(C(C2C=CCS2)=O)CCC1(C)C c1(CNCCNC(c2cccc(F)c2F)=O)cc(F)ccc1Br c1(C(=O)NCCC(C)NC(C2(C)COCC2(F)F)=O)cc2n(n1)CCCC2 Cn1nc(CC(=O)NC2CC(C(CO)NC(C3CCCO3)=O)C2)cc1C(F)(F)F C1(C(N(CC(C)O)Cc2cn(-c3ccc(OC)cc3)nn2)=O)CC(C2CCC2)C1 C1(CCOC)(NC(=O)CCCC2(C)N=N2)CCN(C(c2n[nH]c(=N)s2)=O)C1 C(=O)(C1=C(C)CCCC1)NC1(CCOC)CCN(C(=O)CC2CCNC(=O)C2)C1 C(=O)(CCCC(=O)c1cccs1)N1C(C)CCC1C(=O)NOCC1CCCCC1 C1(C(C)(C)C)(CNC(c2occc2C2CC2)=O)CCN(C(C2CCSCC2)=O)C1 CC(CS(C)(=O)=O)C(=O)N(C(C)CCNC(c1n[nH]c2c1COC2)=O)C c1(C(=O)NC2CC(C)N(C(c3cccc(F)c3F)=O)C2)cc2cc[nH]c(=O)c2s1 N1(C(CC2(C)CCCO2)=O)CC2C(CNC(=O)CCc3ccccn3)C2C1 C1(CNC(c2c(C)cco2)=O)CC12CCN(C(=O)CC1(C)CCS(=O)(=O)N1)CC2 c1(C(N2C(C)C(NC(C3C4CC5C(C4=O)C35)=O)CCC2)=O)cnc2n1CCOC2 N1(Cc2c(OC)nccn2)CC(NC(=O)CCCc2cccnc2)C(C#N)C1 c1(C(=O)NCCNC(C=CC)=O)ccc(NC=O)cc1.C1C(C)(C)N1 N1(C(=O)NCC2CCCC2C2CC2)CCC(c2ncc(-c3ccccc3)[nH]2)CC1 c1(NC2(C)CN(C(CSCCCC)=O)C2)cc(COC)nc(Cl)n1 c1(C(N2CCC(NC(=O)Cn3cccn3)(CO)C2)=O)ccc(Cl)c(F)c1F N1(C(=O)NCCc2cc(OC)cc(Cl)c2)CCCC2(CCS(=O)(=O)C2)C1 c1(C(N2CC(F)(C(=O)Nc3n(CC)ncc3)C2)=O)cccn2nnnc12 CC1=C(CNC(=O)C(C2CCN(C(=O)CN(C)C3CC3)C2)F)CCC1 C1(CC(=O)NC(C=C)COC)CC(F)CN1C(C)=O.C(C)(COC)(COC)N c1(C(N(C2CCN(C(=O)Cc3ccno3)C2)C)=O)cc(Br)ccc1F O1NC(=O)C(CC2CC2)CNC(=O)C1.C1(C(=O)OCC)CCCC1 C1(CNC(c2c(C)nco2)=O)CCCC12CCN(C(c1ccsc1C#N)=O)CC2 C(C)(CO)(C(=O)N(CCCCCNC(=O)C(C)NC(C)(C)C)C)OC Cc1cc(Cl)ccc1NNC(=O)Cc1cccc(Cl)c1Cl C1(C(C)O)CCC(NC(=O)CCC2CCCN2C(c2cnco2)=O)CC1 Cc1ccc(C(=O)NC(C(=O)NCCC[Si](C)(C)CC)C(C)C)cc1F C1(CNC(c2ccc(F)cc2)=O)CCCN(C(c2sccc2CO)=O)CC1 C(=O)(C1CCCc2c1ncn2C)NCC(C)NC(c1cc(C#C)cc(F)c1)=O C(c1ccncc1)=C(C)C(=O)NCC(C)CNC(=O)COCC1CCOC1 c1(C(N2CCC(NC(Cc3ccn(CC)n3)=O)CC2)=O)ccc(Cl)cc1C c1(C(=O)NCC2CC(NC(C(CC)C(C)C)=O)C2)ccc(=O)n2c1COCC2 C1(NC2(CC(=O)N(C)C3CC3)CCOCC2)CCC(F)(F)CC1 c1(C(N2C(CN(C)C(c3csc(Cl)n3)=O)CC(F)C2)=O)cncc(Cl)c1Cl CC(=O)C(C)CC(C)C(=O)NCc1ccc(C(=O)NCC2(CCCO)CC2)o1 CCCC(C)(O)C(=O)N1C2CCC(C2)C1CC(=O)NCC1CCCCN1C C1(C2CCCC2)(NC(C2N(C(C(CC)Cl)=O)CC(O)C2)=O)CC1 C=C(F)C1(CC(=O)NC(C)CN(C)C(c2n[nH]c(CC)n2)=O)CCC1 C#CCC(CC(=O)NC(CCOCC)C(C)C)NC(=O)C(C)NC(C)(C)CC c12ccc(c(Cl)c1)NC(=O)C(=O)N2.c1(C(=O)OC(C)(C)C)cc2n(c1)CCC2 c1(CC(=O)NC(CCOC)CNC(=O)Cc2ccco2)ccc(F)c(F)c1 CCC(CC)CCCC(=O)N1CC(CNC(C2(C)CCC(=O)C2)=O)C2(CCC2)C1 C1(C(=O)NCC(CNC(c2cc(CC(C)C)on2)=O)C)COCCOC1 c1(C(N(CCCNC2CC(C#N)C2)CCO)=O)ccc2c[nH]nc2c1 N1(C(c2c(CNC(Cc3ccc(C)nc3)=O)ccs2)=O)CCC2C(O)C(C)(C)C12 c1(CC)ncc(C(=O)NCC(C)(CNC(c2ccccc2OC)=O)OC)cn1 N1(C(CC(CC=C)(C)C)=O)C2CCC1C(F)C(NC(=O)C(F)C(C)(F)F)C2 C1(CC(N2C(CC(=O)OC)CCC2)=O)CCC(=O)NC1.C12CC1CNC2=O c1(C(=O)NC2C(NC(c3csc(Cl)c3)=O)C2)ccccc1Oc1ccccc1 N1(C(C(CCC)O)=O)CCC(CNC(c2cccnc2OC)=O)C(C)C1 N1(C(C=CC(=O)OC)=O)CCC(C(C)NC(c2cccnc2N(C)C)=O)CC1 C1(C)(C(=O)NCC(C)(CNC(C2CCC(C(N)=O)O2)=O)OC)CC(C#N)C1 C(c1cn[nH]c1)=C(C)C(=O)NCCC1(C(=O)OC(C(C)(C)C(C)C)=O)CC1 Cc1cc(C(=O)NC2CC2NC(C2(C#N)CC3CC3C2)=O)cc(C(F)F)c1 c1(C(=O)NCC=CCNC(Cn2c(C)nnn2)=O)c(C(F)F)nc2ncccn12 n1(CC)c(=O)sc2c(N3CCOCC(C(=O)NCCO)C3)ncnc12 C(=O)(CC(C)C(=O)N1CC2CC1(CNC(C1CCC(F)CC1)=O)C2)OCC c1(C(=O)NC(C(C)NC(C=CC)=O)C)cnn2c(C(F)(F)F)cc(C)nc12 c1(C(N2C(CNC(CCC(=O)NCCC)=O)CC2)=O)cc2cc(F)ccc2cn1 N1(C(C(C(C)C)SC)=O)CCCC(C(N2CCC(OC3CCC3)C2)=O)C1CC C1(C(N2CCC(CCNC(CC(C)C)=O)C(F)(F)C2)=O)COc2ccccc2C1 c1(C(N(CC(CNC(CSCC)=O)O)C)=O)sc2nc(C)nc(C)c2c1C N(C1COc2cc(Br)ccc21)C(=O)Nc1cccc(SC)c1 C1(OC)CC(NC(C2OCCC2C)=O)CN(C(c2csnn2)=O)C1 N1(C(C2(OC)CCCC2)=O)CC2CCC1CN(C(c1ccncc1N(C)C)=O)C2 C=CCCCC(=O)NC1CC1NC(c1cn(CC(N)=O)nn1)=O c1(-c2ccccc2)noc2c1CN(CC1CCc3nccn3C1)CC2 C1(C(N2CCC(C(=O)NC3CC(CC)C3)(CC)C2)=O)CC(=O)NC(C)C1 C#CC1(C(=O)NCc2cncc(C(=O)NC3CN(C)CC3C)c2)CC(=O)C1 C1(NC(CCOCC)=O)C2CN(C(C3(C)COC(=O)C3)=O)CC12 Cc1ccc(S(C)(=O)=O)cc1NC(=O)NCC1=NOC2(CCCNC2)C1 CCC(CC)C(C)C(=O)NCC12CCC(CC1)N2C(=O)C(F)=C1CCC1 C(=O)(C(C#N)C(C)(C)C)NCc1cc(C(N2C(C(CC)O)CCCC2)=O)ncc1 CCCCS(=O)(=O)NC(C1(C)CCN1C(=O)NC(=O)C(Cl)(Cl)Cl)=O C1(NC(C2CCC(C(C)C)CC2)=O)CC2CCC(C1)N2C(C1CC1(C)C)=O N1(C(C2C(C)(C)C2C#N)=O)CCn2ccnc2C1.C1(CN)OC(=O)CC1(C)C Cc1cc(Cl)nc(Cl)c1CNC1CC(CC(=O)Nc2cnccc2C(N)=O)C1 C=CCCC(C)(C)C(=O)NC(C1CCOC1)CNC(=O)Cc1ccn(C(C)C)n1 c1(C(=O)NCc2ccccc2)ccnc2ncnn12.CCC1CNC(=O)C(C)O1 C1(NC(COC)=O)CC(CNC(c2ccccc2SC(F)F)=O)C1(C)C S(=O)(=O)(c1ccccc1)N1C(C(N(c2ccc(C)cc2)CC(C)C)=O)CCC1 c1(C(N2CCC(CN(C)C(C3COC(=O)C3)=O)C2)=O)ccc(F)c(CO)c1 C1(C(C)(C)OC)CCC(C(=O)OC(c2ccc(C(F)(F)F)nc2)C)CC1 N1(C(Cc2cncc(C)n2)=O)CCC(C)C(C(N2CCCC(C(N)=O)C2)=O)C1 C12(NC(c3cnc(CN)[nH]3)=O)CCCC1CN(CCn1ncc3ccccc13)C2 C1(NC(C(Br)=C(C)C)=O)CN(C(c2ccc(F)cc2F)=O)C2CCCCC12 c1(C(N(CC(CC)NC(=O)C=Cc2ccsc2)CC)=O)ccc(-c2cccs2)o1 N1(C(C2CC(OC)C2)=O)CC(C)(C)CCC1CNC(C1CC2(CSC2)C1)=O c12cccc(c1)CNC(=O)NC2.c1(C(=O)OCC)ncc(C(C)(C)C)s1 CCCCC(O)C(C)C(=O)NCc1cnn(C)c1C(=O)NOCc1ccccc1F C1(NC(C#CCNC(C2OCCN(C)C2)=O)=O)CCCC(F)(F)C1 c1(CC(N2C3C(NC(CCCC(C)C)=O)CC(C3)C2)=O)ccccc1S(C)(=O)=O C1(C2CCOCC2)(CNC(C=C(C)Cl)=O)CCN(C(=O)CNC=O)C1 C(CCC(C)C(=O)NCc1cc(C(=O)NC2CC3(CC3)C2)ccn1)OC C(c1cn[nH]c1)=C(C)C(=O)N(CCC(C)NC(=O)C(F)F)C N1(C(CCC(=O)OC)=O)CC2CCC(C1CO)N2C(c1cc(C)c(F)c(C)c1)=O Cc1nccc(C(=O)NCc2ccc(C(N3CCC4CC4C3)=O)s2)c1N c1(N(C(=O)NC2CC(COC(C)=O)C2)Cc2nc[nH]n2)c(C)cc(C)cc1C.CO N1(C(C2C(C)N(C)CC2)=O)CC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2C1 c1(C(N(C2CCN(C(=O)CSCC(=O)OC)C2)CCC)=O)n[nH]c(C)c1C C(C(=O)NCC(c1ccccc1)NC(=O)Cc1ccc(C)nc1)(C(C)C)NC(C)=O C1(C(=O)NC(c2ccccc2-n2ccnc2)C)CCNC12COC2 CC1(F)CC(C(=O)N(CCCNC(=O)CC2CCCO2)CC2CCCCC2)C1 c1(CC(N2CC(C)C(NC(C3CN4CCC3CC4)=O)C2)=O)cccc2[nH]ncc12 C1(CNC(C2(CCNC(c3ccn(CCF)n3)=O)CC2)=O)CCC(=O)N1 c1(C(N2CCCC(Cc3cn(CCCC)nn3)C2)=O)cc([N+](=O)[O-])cnc1O C1(CC)(CNC(c2ccc(C(=O)NC(CO)CCOC)[nH]2)=O)CC(C)(C)C1 N1(C(C(=O)NCCOCCCC)=O)CC(CO)C2(C1)CN(C(C1CC1C#N)=O)C2 c1(C(N2CCC(C)(NC(=O)CC3CCOCC3)C2)=O)cnc2c(c1)CNC(=O)N2 c1(C(N2C(CC(=O)NC(c3cncnc3)C)COCC2)=O)ccc(Cl)c(C#N)c1 C1(CC)C(NC(c2cnco2)=O)CCN1C(=O)CCOCC(C)C C1(C(N2CCC(CN(C(c3cc(C)sc3)=O)C)C2)=O)CC(F)(F)CS1 C(=O)(C1=CC2CC(C1)CC2O)NCC(CCCC)NC(c1[nH]cc(C)c1C)=O c1(N2CCC(NC(C3CCC4(CCC4)CO3)=O)C2)ncnc2c1CCC2 c1(C(=O)NC2(C(=O)OC)C(CNC(COCCC)=O)C2)c(C)cc(O)nc1C CCCCCC(CC)C(=O)N(CCN1CCN(C(=O)C=CC2CC2)CC1)C1CC1 c1(C(=O)NCC2OCCC(NC(CCOC)=O)C2)cnn2cc[nH]c(=O)c12 N1(C(c2cn(CC=C)nc2)=O)CCCCC1CN(C(=O)CC(C)c1ccco1)C N1(C(CCCCSC)=O)CCC2CC1CN(C(c1sc(C(F)(F)F)nc1C)=O)C2 CC(CCC(=O)NC1CCN(C(c2cc(C3CC3)nn2C)=O)C1C1CC1)N(C)C C1(S(N)(=O)=O)(C(=O)NC2CCN(C(c3c(C)cc(CO)o3)=O)C2)CCCC1 C(N=c1nc2c(cnn2C)c(N2CCOCC2)[nH]1)c1n(CC)nnn1 c1(C(=O)NC(CNC(C(C)(C)SC)=O)C2CC2)ccc2c(c1)nnn2C C1(C(=O)NCC23CC(NC(C(CCC)OC)=O)(C2)C3)CC2CC2CC1C c1(N2CCN(C(c3ccc(C)nc3C)=O)C3C2C3)ccnc2ccnn12 N1(C(C2(CNC(C=CCC)=O)CC=CC2)=O)CCSC2CCCC12 N1(C(c2cc(C)cc(Br)c2)=O)CC2CN(C(=O)C=Cc3ccc(O)cc3)CC2C1 c1(C(N2C(C)CC(NC(=O)C=CC3CCCO3)C2)=O)cc(F)cc2nn[nH]c12 n1(CCOC)nnnc1C(C(C)CSc1ccccc1)NC(=O)OC(C)(C)C N1(C(CCCOCC=C)=O)CC2C(CNC(=O)CCN3CCC3)C2C1 CC1=C(C(=O)N(C2CN(C(c3nonc3N)=O)C2)C)C=C2CCCN=C2N1 N1(C(C(CCOC)C)=O)CC2CC(CNC(=O)C(c3ccncc3)C)C2C1 C1(C(N(CC(=O)NCCCCCCO)CC)=O)CCN2CCCC2C1 CC(CC(=O)NCC(C)(C1CC1)NC(=O)CNC(N)=O)n1cc(Br)cn1 C=CC1(CC(N2CCC(C)C(NC(C3COC4COCC34)=O)C2)=O)CCCCC1 C(=O)(C=C1SCC(=O)N1C)NC1(COC)CCN(C(c2cnc(CCC)s2)=O)C1 CC(C)(C(=O)N1CCC(C(N)=O)C1)NC(c1coc(C(N)=O)c1)=O C(CCS(C)=O)(C(=O)NCCNC(=O)CCCc1cccs1)N(C)C C1(NC(C2C(OCC)C2)=O)CCC1NC(=O)Cc1cscn1 C(CCO)(C(C)(C)C)NC(C1CC(NC(CC2CCN(C)C2)=O)C(O)C1)=O C=CCC(C(=O)NC1(C(=O)NC(CC)C(C)(C)O)CCCCC1)OC N1(C(C(C)(C)SC)=O)CCC(C2CCCN2C(c2ccc(C(C)C)s2)=O)CC1 c1(OCC)ccc(C(=O)N(C2(CNC(C3CN(S(C)(=O)=O)C3)=O)CC2)C)cn1 C(=O)(CCCC(=O)N1CC2C(C(=O)NCC(C)(C)C(C)O)C2C1)OC c1(OC(C)C)ccc(C(C(=O)NC2CCCO2)N(CC(C)C)CC)nn1.C(C)(C)(C)O N1(C(CCN(C)CC)=O)CCN(C(c2cc(-c3ccn(C)n3)on2)=O)CC1CO S(=O)(=O)(c1cc(F)ccc1F)N1CC2CN(C(=O)CC3CC3)CC2C1 N1(C(CNC(=O)OCC=C)=O)CC(C)CN(C(C2(F)CCC2)=O)C(C)C1 N#CC1(CCN2CC(CC(F)C=O)C2)CCOC1.N1CCC(N2CCC2)CC1 Cc1oc(C(N2CCC2CNC(c2ccc(CO)cc2)=O)=O)cc1S(C)(=O)=O c1(C(=O)NCCC(C(C)C)NC(=O)CCC2CCCCC2)ccc2ccnn2c1 N1(C(C2C(C)CC2)=O)CCCC(CNC(c2csnn2)=O)C1 c12ncc(cn1)c(=O)[nH]2.c1(N(C2CCN(CC)C2)C)nccc(C(C)C)n1 c1(C(=O)NC2CN(C(Cc3ccc(C)nc3)=O)C2)ccc(C(F)(F)F)nc1O C1(C(N(C2CC(C(N)=O)C2)C)=O)(NC(c2ccncn2)=O)CCN(C)C1 C=CCCCCC(=O)N1CCCN(C(=O)C=Cc2c(C)noc2C)CC1 C1(C(=O)NCC2COCC3(CCN3C(=O)OC(C)(C)C)O2)CNC(=O)CC1CC C(C(C(=O)N(C)Cc1cnn(C)c1)NC(=O)CCn1ccnc1C)OCC C1(OCC)CN(C(=O)C=CSCc2ccco2)CC1NC(c1ccc(=O)oc1)=O c1(NC(C2(C#N)CC3CC3C2)=O)c(Cl)sc2nnsc12 C1(NC(COCCc2n(C)cnc2)=O)CCC2CN(Cc3ccccc3)CC2C1 C1(CN(C(C(CC)=CCCC)=O)C)CCCN(C(c2cncc(C)c2)=O)C1 C1(CNC(C2C(C3C(C)C3)C2)=O)CC2(CO1)CN(C(C1(C)COC1)=O)C2 c1(C(N2CC(N(C(=O)CSC(C)(C)C)C)C(F)C2)=O)csc2ccccc12 c1(C(=O)NCC(CCCC)NC(=O)Cc2csc(S)n2)cc[nH]c2nccc1-2 CC1=CC=CNC(=O)NCC1CCN1CC(OCCCO)C1=O C1(COC(c2c(CC)c[nH]n2)=O)CCC2COCCC2C1 CCC(C)(C)CCCC(=O)N1CCN(C(c2nc(C)ccc2F)=O)C2CC12 N1(C(C(CCOC)C)=O)CC(NC(=O)C2=CSCS2)CC(F)C1 c1(C(N(C(CNC(C2CC3CC3C2)=O)C2CC2)C)=O)csc(O)n1 c1(-n2cc(CNC(CNC(=O)NC)=O)nn2)cccc(C(=O)NC2CC2(Cl)Cl)c1 N1(C(N2CCN(CCc3ccccc3)CC2)=O)CCCC(CF)C1 C1(C(=O)NCc2occ(C(N(C)Cc3ccncc3F)=O)n2)CC2C=CC1CC2 N1(C=O)CC2CC2(CNC(c2ccnc(N3CCCC3)c2)=O)C1.CC(C)(F)CC c1(OC)ccc(CC(=O)N(C(C)CNC(C2(CF)CC2)=O)C)c(Cl)c1 C(C1CCOc2ccccc21)OC(C1C(OC)CN(C(=O)OC(C)(C)C)C1)=O C1(OC)CC(CF)N(C(=O)CN(C(C2CC(O)C(F)C2)=O)CC2CC2)C1 c1(C(N(C)CC2N(C(CCC3CC(C)C3)=O)CCOC2)=O)c2c(nn1C)CCC2 N1(C(C2C(C)C2)=O)CCC(CNC(c2cc3sccc3n2C)=O)C(F)(F)CC1 c1(C(=O)Nc2cccc(C3CCCCC3)c2)cc2cc(Cl)c(Cl)cc2[nH]1 C1(CNC(C2N(CC)CC2)=O)CCC(F)CC1.C12(OC)CN(C1)C2=O c1(C(N2C(C(=O)NCC3(O)CCC(C)C3)C(O)CC2)=O)c[nH]c2ccncc12 Cc1ccc2ncc(C(=O)N(C)CCN(C(=O)CC(C)N3CCCC3=O)C)n2c1 N1(C(C(c2cccs2)N(C2CC2)CC)=O)CC2CC2(C(CNC(C2C(C)C2)=O)=O)C1 C(C(O)CN=c1ccnc(C2CCCC2)[nH]1)NC(C=CC=CCC)=O c1(NC(=O)Nc2scc(C(CC)C)n2)ccccc1S(=O)C(F)(F)F C1(C(N(CC=C)CCOC)=O)CN(C(=O)C(C2CCCCC2)O)CC1C N1(C(CCN(C(C)=O)C)=O)CCOC(C)(CNC(=O)C(C)CN(C)C)C1 CC1CCc2ncc(C(N3CCCC(N(C(=O)Cn4cnnc4O)C)C3)=O)n2C1 NS(=O)(=O)CCCCCCC(=O)NCC1(C(=O)NC2CCCCC2)CC1 Cc1oc(C)c(C(N2CCCCC(NC(=O)C(CCO)N(C)C)C2)=O)c1C C1(C(=O)NCC(=O)OC(C)C)CCCN(C(=O)CC2CCCOCC2)CC1 S(=O)(=O)(c1ccc(=NCc2c(C)noc2C)[nH]c1)N(C(COC)(C)C)C CCCCC(O)CC(=O)NC(C)(C)CC(=O)NC(c1ccoc1)C C=CC(CCC)CC(=O)N(C1CCC(CNC(=O)C(C)C2(O)CCC2)CC1)C C1(CC(=O)NCC2(CN(C)C(c3ccncc3)=O)CC2)CCC2(CC2)CO1 N1(C(C)=O)CCOCC1CC(=O)NC1CCCCC1NC(=O)CSC(F)(F)F CC(C)(C)C(CCNC(c1nnn2c1CSCC2)c1nnnn1C1CC1)C(F)F CC1CCC=C1C(=O)NC1(C)CC(NC(=O)CCF)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCN(C(c1c(CCC)cccc1)=O)C1CC1 C1(C(c2nnnn2C)Nc2sc(Cl)nc2C)(OC)CCCN(C(C)(C)C)C1 C1(C)(C(=O)NC(C2(O)CN(C(COc3cc(C)on3)=O)C2)C)CCC(=O)NC1 c1(C(N2CC(CCNC(C3CCCC3c3ccccc3)=O)C2)=O)csc(O)n1 c1(C(=O)NC(c2occ(C(N(C3CCC(C)C3)C)=O)n2)C)ccccc1O c1(C(N2C3CN(C(CCCC(=O)OC)=O)C(CC3)C2)=O)cnc2ccccc2c1 C(C1c2ccccc2OCC1NC(=O)OC(C)(C)C)N(Cc1cn(C)nn1)CCO C12(C(=O)NC3CCN(C(=O)NCC)CC3)CCCC1(F)CN(C(=O)C(C)CO)C2 c1(C(=O)NC2C(NC(C3(NC(CSCC(C)C)=O)CC3)=O)C2)ccsc1 c1(C(CC(C)NC(C(C2(O)CN(C(C)=O)C2)O)=O)O)ccc(F)cc1F CC1CCC(NC(C2CSCN2C)=O)CN1C(=O)CC1CCN(C)C1=O C(=O)(C1=CC2(CCN(C(c3csnc3C)=O)C2)C1)N1CC(C(CC)C)C1 C(=O)(CCCC(=O)NCC1(NC(=O)COC2CCOC2)CCOC1)OCC C(=O)(C(C)CS(C)(=O)=O)NC1CC2(C(NC(c3c(C)nc(CC4CC4)o3)=O)C2)C1 C(C(CO)N=c1nc2[nH][nH]cc-2c(O)n1)NC(=O)CCC1CC1(F)F N(C1CCCOc2ccc(Br)cc21)c1ccc2nc(O)n(C)c2c1 c1(CCC)nc(C(=O)NC(C2CCN(C(=O)CCc3cc(C)on3)C2)C)cs1 c1(C(=O)NC(CN(C(CN(C2CC2)CC)=O)C)C)n[nH]cc1F C1(C(=O)NCCc2n(C)ncc2)CC12CCN(C(=O)C(=O)NCC1CC1)C2 C1(NC(c2cccc(OC)n2)=O)CC12CCN(C(=O)CC(C)C(C)C)C2 CC1(C)CCC(C(N2CCC(NC(c3ccc(CC#N)cc3)=O)C2)=O)O1 Cc1cc2cc(C(=O)NCc3ccc(OC(F)(F)C(F)(F)F)cc3)ccc2s1 N1(C(c2cnn(C(C)C)c2I)C(=O)NCc2cccs2)CCC(C)(C)C1C N1(C(C(CCC)N(C)C)=O)CC(NC(c2cnc(CCC)s2)=O)CC1(C)C Cc1cc2ncc(C(=O)NCC34CC(CO3)N(C(C3CCC(C)O3)=O)C4)cc2[nH]1 C1(C(N2C(CN(C(=O)Cc3cnsc3)C)COCC2)=O)CC2CC1C1C2C1(F)F CCC(CC)(CO)C(=O)N1CC=CC(NC(=O)C(=Cc2cscn2)F)C1 c1(C(=O)OC)nccc(N(CC(C)NC(=O)C(n2nc(C)cc2C)C)C)n1 C(=O)(C(F)C(C)(F)F)NC(C1CC=CCC1)C(=O)NCCN(CCO)CC c1(CC)ncc(C(N2CCOC(C)(CNC(=O)C(O)C(F)(F)F)C2)=O)c(O)n1 C1CN=C2C=C(N=C(Cl)N2)O1.Cc1noc(Cl)c1CCC(=O)NCCOC(C)C C(=O)(C1=CSCCO1)N1C(CCNC(c2ccn(CC)c2C)=O)CCCC1 C1(CC)CN(C(C2(COC)CN(C(=O)C3=COCCC3)C2)=O)CC12CC2 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(C(=O)C(C)n2ccnn2)CC1)C N1(C(CCCCC#C)=O)CCC(CNC(=O)CCN2CCC(F)C2)C(F)(F)C1 c1(C(=O)NCCOCCCC)ccc(CNC(C2CC(CCO)C2)=O)s1 Cc1cc(C(N2CC(NC(C3CC3(Cl)Cl)=O)C(C)(C)C2)=O)c(N)cc1F c12cc3c(s1)CCN(C3)CCOCC(C)n1c-2nc(CSC(C)(C)C)n1.CCS.CC C1(NC(C=CSC)=O)CCN(C(=O)CC2C(=O)ON=C2C)C1C c1(C(N2CC(S(CC)(=O)=O)C2)=O)ccc2c(c1)SCC(=O)N2 C(=O)(C(C)(C)Cc1cccc(Cl)c1)NCC(C)CNC(=O)CC1C=CCCC1 c1(SC)ncc(C(=O)NC(CO)C(C)NC(C2C(C)(C)C2(F)F)=O)c(O)n1 C(c1cnccn1)=CC(=O)NCC(CNC(c1ncnn1C(C)C)=O)OC c1(C(N2CC(NC(C3CSC3)=O)(CO)C2)=O)ccc(Cl)cc1Br N(C1CCc2cc(CNC(c3ncsc3C(F)(F)F)=O)ccc21)C(C1C(C)C1)=O Cc1c(F)ccc(CN2CCC(O)(CC(=O)Nc3nc(Cl)ccc3Br)CC2)c1Cl N1(C(C2C(C(=O)O)CC(c3ccccc3)C2)=O)CCC(O)C12CC2 c1(C(N(C2CN(C(c3cc(Br)no3)=O)C2)C)=O)cc2ccccc2s1 N1(C(Cc2c(C)con2)=O)CCCCC(CNC(=O)CCC2CCCCO2)C1 c1(C(=O)NCC(CN(CCCOCC)C)(C)C)c(OC)cc(Br)cc1F C(N=c1nc(O)c2cnn(C)c2[nH]1)C1(O)CCN(C(C(COC)(C)OC)=O)C1 N1(C(=O)OC(C)(C)C)CC2(CCC2OC2CC23CC(C(=O)ON)C3)C1 N12CC(NC(C=CC=CC)=O)CC1C2.C1(=O)CS(=O)(=O)NCCN1.C(C)=O CC1(C)OCCNC1C(N1CCN(S(=O)(=O)CO)CC1)=O O=S(=O)(c1ccc(Cl)cc1F)NCc1c[nH]c(=NCc2ccc3ccoc3c2)s1 c1(CNC(=O)CN2CC3CCCC3C2)ncnc2[nH]ccc12.c12ccccc1S2 C1(C(=O)NCC(C)NC(=O)C(C)c2ccon2)CCN(C)C(=O)C1 c1(OC)ccc(CN2CCCC(C)(C(N3CCOC(CO)C3)=O)C2)c(OC)c1C C1(CC)CC(C(=O)N(C)CC2CC(O)C2)CCN1C(c1cc(C)cs1)=O C1(C(=O)NC(N)=O)(NC(C(CO)N(C(=O)CN2CC3CCC2C3)C)=O)CCCCC1 Cn1nc(C(N2CCCC(CO)(NC(=O)C(C3CCOCC3)F)C2)=O)cc1C#N N1(C(C(C)OCC#C)=O)CC(C)(C)CC1C(=O)NCc1nonc1CC c1(C(=O)NC(CCOC)CN(C)C)c(C(=O)OC)c(C(F)(F)F)nn1C CCC(F)(F)C(C)(C)C(=O)NCC1(C)CN(C(=O)COC2CCOC2)C(C)(C)C1 C(=O)(C1=CC2CCC(C1)C2)NCCN.N1(CC(C(=O)CC2CCCC2)=O)CC2CC2C1 C(=O)(CC1CCc2ccccc21)N1CCC(N(C(COC(C)=O)=O)CC2CC2)C1 C1C(CC2CC2)C(=O)N1.C1(CNC(COCC(C)C)=O)CCOC1C(C)C Cc1cc(NC2CCC(=O)NC2C)n2nc(C)nc2n1 C(C1CC(=O)Nc2ccccc21)Nc1ccc(C(=O)OCC(N)=O)cc1 c1(OC)ncc(C)cc1NC(C1CC=CC(NC(C2CNC(=O)O2)=O)C1)=O c1(C(N2CC(NC(c3c(CC)[nH]cc3)=O)C(C)C2)=O)cc2c(Cl)cccc2[nH]1 c1(C(=O)OC)cc2c(N(C3CCCC34CC4)C3CC3)nccc2s1 Cc1cc(-n2nc(-c3cncs3)nc2CC2CCCN2C)cc(C)n1 CC12CCCN(C(=O)C(N3CCNC4(CCC4)C3)=O)C1COC2 C1(C(=O)NCc2ccc(C#N)s2)(CC)CCN(C(=O)CC2CC2C)CC1 C1(C(=O)NC(C#C)CCC)CC(O)C(O)CC1CNC(=O)CC(C)C(=O)OC N1(C(C2C(C=CC)CN(C(=O)CCCCCOC)C2)=O)CC2CCC1C(O)C2O CC(C)(CNC(=O)CN1CC2CC2C1)CCNC(=O)COc1ccccc1Cl c1(N2CC(CNC(Cc3c(C)cncc3)=O)OCC2)nc(C2CC2)nc(=N)[nH]1 C1(CN(C)C(c2cc[nH]c(=N)c2)=O)C2CN(C(=O)C(C)(C)c3nccn3C)CC12 C1(OC)CC(C(=O)NCCNC(=O)CC2CCC(=O)C2)N(C(=O)C2CC2)C1 N1(C(CC(CC)OC)=O)CCC2(CC1)CC2CNC(C1(C(=O)N(C)C)CC1)=O C(=O)(C(CNC(C1CCOC(C)(C)C1)=O)C(C)(C)C)N(CCN1CC=CC1)CC c1(C(N2CCN(C(C(CC=C)C)=O)C(CCC)C2)=O)cc(S(N)(=O)=O)oc1C N1(C(C2(CC=C)CC2)=O)CC2ON=C(CNC(C3(Br)CC3)=O)C2C1 N1(C(c2ccnn2CC(F)(F)F)C(=O)NCC(F)F)CCOC2CCCC12 n12nc(C(F)(F)F)c-1c2C.C1(CNC(C)=O)COCCN(C(=O)C(C)(C)CF)C1 C1(CC)CN(C(C2(OC)CCOCC2)=O)CCN1C(c1csc(Cl)n1)=O C(N=c1cc(C#N)[nH]c2ccccc12)c1ccc(OCC=C)cc1 N1(CC(=O)NCC2CCCC2NC(c2ccc(=O)oc2)=O)C(=O)CCCC1=O C1(CNC(CSCC#C)=O)(OC)CCN(C(=O)CC2CCOC2(C)C)CC1 N1(C(C2(SC)CC2)=O)CC(CNC(=O)C(C)Oc2ccc(C#N)cc2)C2(CC2)C1 CCCCC(C)C(=O)N1CC(NC(c2cc(N)cnc2Cl)=O)C(C)C1 c1(C(=O)NC2CN(C(C3CN(C)C3)=O)CC2O)cccc2c1oc1ccccc21 N1(C(Cc2n(C)nnc2)=O)CC=C(C(=O)NC2C=CCC2)CC1 c1(C(N2CC(O)(CCNC(C(CO)OC)=O)C2)=O)cnn(C(C)C)c1C CCS(=O)(=O)C=CC(=O)NC1CCC(CNC(c2cc(C(N)=O)[nH]n2)=O)C1 c1(C(=O)NC2C(C)CCN(C(CC(C)C)=O)C2)nc(=N)[nH]c2ccccc12 C(c1ccc2nc(C)oc2c1)=CCn1c(=O)ccc(C)n1 Cc1cc(C)c(NC(C2(C)CC(NC(C3CCCN(C)C3)=O)C2)=O)cc1O c1(CC(=O)OCC(C)(C)OC(C)=O)ccccc1.C1(C(=O)N)CC1C(N)=O N1(Cc2cn(C(CCC=C)C)nn2)CCc2cc(C)cc(C)c21 C1(CC)C(C(=O)NC(c2ccnn2C)C)CCN1C(=O)C(CCOC)OC N1(C(CS(CC)=O)=O)CCCC2(NC(=O)C(c3ccc(Cl)cc3)C)CC2C1 N1(C(CC(=C)C)=O)CC2CCC1CN2C(=O)C(c1c(C)noc1C)C C1(C(=O)NC(C(C)C)CN(C)C)CCCN1NC(=O)CCC(N)=O C(=O)(CCN=C(NCC(C(C)(F)F)c1ccccc1)NC1CC1OC)NC N1(C(CCc2cc(C)on2)=O)CCC(F)(CNC(C2C3COCC23)=O)CC1 C1(NC(=O)Cc2ccc(Cl)cc2F)CC2CN(C(=O)COC(F)F)CC2C1 C1(CCC)(C(=O)NCC2CC(C)N(C(c3csc(Cl)n3)=O)C2)CCNC1=O Nc1cc(C(=O)NCC2CC2NC(c2ncoc2-c2ccon2)=O)nc(O)c1 C1(NC(c2c(CC)nco2)=O)CC2CC(C1)N(C(=O)CC1CC(C)(C)C1)C2 C1(NC(C(=Cc2ccc(F)cc2)C)=O)CC2CCC(C1C)N2C(C1CC(=O)N1)=O N1(C(c2c(CC)[nH]c(=N)s2)=O)CCn2nc(C)c(CNC(c3cnns3)=O)c2C1 CC1(C)NC(=O)CC1C(=O)NCC1(NC(c2cnc(C(N)=O)s2)=O)CCCC1 c1(N(C(C)C(=O)OC2CC(F)(F)C2)CC)cccc(CCC(C)C)c1 c1(C(c2cccc(C(=O)O)c2)=O)cc([N+](=O)[O-])cnc1O N1(C(CC2C(C)CC2)=O)CCC(C2(O)CN(C(=O)C=CCn3cncn3)C2)CC1 N1(C(c2cc(CC)oc2C)=O)CC2CCC(NC(C3CCCCS3)=O)CC2C1 CC1C(NC(=O)Cc2cn3ccsc3n2)CCCN1C(C1CC(N(C)C)C1)=O C1(F)(CC(=O)Nc2ccc(C)nn2)CN(C(=O)Nc2ccccc2)CC1C1CC1 N1(C(C=C(CC)CC)=O)CCCC(C)(C(N2CCC2CN=[N+]=[N-])=O)C1 c1(C(N2C3C(NC(C=C(C)C)=O)CC(C3)C2)=O)cc(C)cc2ccncc12 C12(CCCC1)c1cn(nn1)C(C)C(=O)N2.C1(C(=O)NC(COC)C)CCCCC1 CCCCC(CNC(C1CCCCN1C)=O)NC(=O)CC1CCCC1C N1(C(C(CCC)C)=O)CC(NC(c2ccccc2OC2CC2)=O)CC2(CCC2)C1 Cc1cc(C(N2CCC3CC2CN(C(C2(CO)CCC2)=O)C3)=O)cc2nc[nH]c12 CC(C)CC(C(=O)N1CCC=C(Cl)C1)ONC(c1cccc(F)c1)=O C1(NC(CC2(CC)CCOCC2)=O)CN(C(c2cccnc2O)=O)CCC1C Cc1cc(C(=O)NCC(C)(C)CC2CN(C(C3CCC(N(C)C)C3)=O)C2)oc1C C(=O)(C(C)(C)C(C)(F)F)NCC1CC(C)N(C(=O)CCC2CCCC2)C1 CC1CCN(C(C23CCC2CC3)=O)C(CNC(=O)COCC2CCCO2)C1 c1(CC)cc(C(=O)NC2(CNC(C3COC(=O)O3)=O)CCCC2)ccc1OC N1(Cc2ccc(C)c(F)c2)CCc2ccc(NC(C3CCC(=O)N3)=O)cc2C1 c1(C(=O)Nc2cnsc2)cc(C)nc2onc(C)c12.C12(OC)CCN(CC1)C2 N1(C(CC(C)(C)C#N)=O)CC(F)(F)CC1(C)CNC(=O)CC1CC2(CCC2)CO1 N1(C(CCCC=C)=O)CCC(C)C(CC(=O)N(C)CCSC)C1 C1(C(N(CCO)CC2C(C)C2)=O)CCC(F)(NC(=O)OC(C)(C)C)C1 C1(COc2ncc(C(N(CC)CC)=O)s2)CCN(c2nccc(Cl)n2)CC1 C1(CNCc2cn(C3C(OCC)COC3)nn2)CC(=O)N(c2cnn(C)c2)C1 C1(NC(CCOCC)=O)CC2CCC1(C(=O)N(CC(=O)OC)C1CC1)C2 CN(CCCC(=O)NC1C=CCCC1NC(C1(NC(N)=O)CC1)=O)N=O c1(COCCOC)nc(C(N2CCC(CCNC(C3CC3CC)=O)C2)=O)co1 Cc1csc2cc(C(=O)N(C3CN(C(=O)CC(C)(C)CC(F)F)C3)C)[nH]c12 CC1CCN(C(=O)C(C)(C)C#N)CC1NC(=O)CC1CCCCC1 c1(C(=O)NCC2CN(C(C3(C(C)OC)CC(=C)C3)=O)C2)ncc(C)cc1F C1(CC(=O)NC2CCN(C(C)=O)C2)C2CCCC2N1C(c1cccc(N)c1)=O c1(NCC)scnc1C(=O)NC(C)CNC(C12CCC1C2)=O C1(C(=O)NCCC(C)NC(COCC)=O)CCCC(=O)CC1 N1(C(Cc2c(C)noc2)=O)CCC(C)C(NC(=O)CCc2ccncc2)C1 Cc1ccc(Cl)cc1OCC(=O)NC1CCC(C)N(C(=O)CC2CC(F)C2)C1 n1(CC(=O)N(CCC(=O)NC(c2cnc[nH]2)CO)CCO)ncccc1=O Cc1nn(CC(=O)NCC(CNC(C2(CC(C)C)CCC2)=O)CO)cc1Cl CCCCCC(=O)NCC(=O)NCCN(C(=O)CC1COCC(C)O1)C(C)C N1(C(c2c(C)oc(C3CC3)n2)=O)CC(CNC(C2(C3CC3)CC2)=O)C(F)(F)C1 C=CC1CN(CC2CCCC(NCc3ccccn3)C2)CC1O C1(C(N2CCC(O)(c3ccc(F)cc3)CC2)=O)C2CCC1N(C(C1(O)CC1)=O)C2 C(=O)(CC(CC(=O)O)c1ccc(Cl)cc1F)OCCSCC.c1(SC)ccc(O)cc1 S(=O)(=O)(c1ccccc1F)N1C(CNC(=O)Cc2c[nH]c3cccnc23)CCC1 Cc1c(NC(C2CC2C)=O)[nH]c2cc(C(=O)Nc3nc(C#N)cs3)ccc12 C12(NC(c3ncccc3O)=O)CCC(NC(C34CSCC3C4(F)F)=O)(CC1)C2 N(C1CCc2ccc(F)c(F)c21)C(c1n(CC(=C)C)nnn1)c1nc(CC)cs1 N1(C(C2(C3CC3)CN(C(C(C(C)(F)F)F)=O)C2)=O)CC2CC=CCC2C1 c1(C(N(C(C)C)CCN(C(=O)CCC2CCCC2)C)=O)ccc2oc(O)nc2c1 C(=O)(C1=CCC(NC(C2(CF)CC2)=O)C1)NCCCC1C(C)C1 C1(NC(c2ccc(Br)cc2)=O)CN(C(C2(CF)CC2)=O)CC1n1cccn1 c1(C(=O)OCC)cc(C)nnc1N(CCCN(C(=O)C1=CCSC1)C)C N1(C(C(OC)OC)=O)CCC2(CCCC2NC(=O)CS(N)(=O)=O)CC1 S(=O)(=O)(c1cc2sc(=NCC(C)CO)[nH]c2cc1Cl)NCCCCCSC C1(C(N(C)C)=O)CCN(C(=O)NCC2C=CCCC2)C1 N1(C(CC(=C)C)=O)CCCC12CCN(C(C1CC(=O)N(c3cnn(C)c3)C1)=O)C2 N1(C(C(F)=C(C)C)=O)CCN(CC2(NC(C3COC(=O)N3)=O)CC2)CC1 c1(CN(C(=O)NC(C(=O)OCC)C)C)ccc(S(=O)(=O)N(C)C(C)C)o1 c1(C(=O)NCCC(=C)CNC(C2(OC)CC3CCC2C3)=O)c(C)ncnc1C N1(C(=O)NCC2(Cc3ccccn3)CCO2)CCC(c2ncc[nH]2)C1 CC1CN(C(=O)CCn2cccn2)CCN1C(=O)CC1CC=CCN1C C1(C(=O)NCC=CC)CCN(C(=O)C(C)(C)n2cncn2)C(C)(C)C1 c1(C(=O)NCC2CCC3(CN(C(C=CCCC)=O)C3)O2)cnn2c1CC(F)(F)C2 C(=O)(C1=CC2CCC(C1)C2)NCC(C(C)C(C)C)NC(CCNC(=O)OCC)=O C(=O)(C(C)(F)C(=O)NCC1(O)CC(CNC(=O)CCCSC)C1)OC Cc1cc(-c2noc(NC(=O)CN3CC(CO)(CO)C3)n2)ccc1F c1(CCCC(=O)NC2(CCNC(=O)CSc3nncs3)CC2)ccc(F)c(F)c1 NC(=O)CC(O)C(=O)NCc1csc(C(N2CCCC(C(N)=O)C2)=O)c1 c1(NC(=O)Nc2cccc(C3OCCO3)c2)ccc(C2CC2)nc1 C12(C(=O)NC3(C)CC3)CC(CO)(C1)OC2(C)C.N12CCC(C1)N(CCO)CC2=O c1(C(=O)NC(CC)CN(C(=O)CSc2nnc(S)s2)C)cc(OC)n(C)n1 Cc1sc2ncnc(C(=O)NC3(C)CCC(NC(C)=O)CC3)c2c1C N1(C(Cc2ccc(CC)s2)=O)CC2OCCCC2(C(=O)OCC(C)(C)C)C1 C(=O)(CCC(CC)OC)NCc1c(C(N(CC#C)CCO)=O)occ1 C(CNC(=O)CSc1ccccc1)(CC(F)(F)F)NC(C1(OCC)CCSC1)=O C(=O)(CCCCC(C)(C)C)NC1CC(CNC(C(C=C=C)C)=O)CC1O c1(C(=O)NC2CN(C(C3CCCS3)=O)CC2F)ccc2nccnc2c1 N1(C(c2c(C)occ2)=O)CCN(C(=O)Cc2nncn2C)C(C)C1C CC(C(=O)NCCC1(O)CCCN(C(c2cnc(C3CC3)o2)=O)C1)C(C)(C)C c1(CNC(=O)Cc2csc(C3CCC3)n2)nc2ccccc2[nH]1.c1nn[nH]n1 c1(C(=O)NCCCCC2C(C)C2)cc2ncn(C)c2cn1 C(=O)(C1CCCc2cncn21)NCc1c(CNC(C2(N(C)C)CC2)=O)cccc1 c1(-c2noc(C)n2)cc(Cl)ccc1F.C(C(=O)NC)NCCCN(C=O)CC C12CCc3nnc(n3C1)NC2.c1(CC#N)ccc(N2CCCCC2)nc1 C1(CCOC)(NC(=O)C=CCO)CCN(C(=O)C(O)CC2CCCCC2)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2(CCC2)CC1CNC(c1cc(Br)n[nH]1)=O C#CCC(C(=O)N1CCCC1(C)CC)NC(C1CS(=O)C1)=O C1(C(=O)NCCC2CC(NC(C3CC4CC4C3)=O)C2)CC2COCC(C1)C2(F)F c1(CC(N2C(C(=O)NC3CC(CC)(CC)C3)CC2)=O)ccc(Br)cc1 c1(CNC(C=C(CC)CC)=O)ccnc(OC)c1.C12(CSC1)C(=O)N2 Cn1ccc2cccc(C(=O)NC3CCCC3C(=O)N(c3ccccn3)CCO)c12 N1(C(=O)OCCC(C)C)CC2CN(C(=O)CCCc3ccc(Cl)cc3)C2C1 C(C(C)(CC(C)C)NC(C1C2CCCC12)=O)NC(CNC(=O)NC)=O N1(C(c2cccc(C(C)C)c2)=O)CCC(NC(c2ncsc2C2CC2)=O)C(F)C1 N12CCC(F)(F)C(C1)C2=O.c1(C(=O)Nc2cncc(Br)n2)cc(O)ccc1O C(=O)(CCC1CCCO1)N(C(C1(CC(=O)OC)CC1)=O)C CC1=C(C(=O)N2CCN(C(=O)C(C)C#N)CC2CC2CCCCC2)CCC1 CCCCC(C(=O)N=c1cc2n([nH]1)CCCC2)NC(=O)C(CO)C(C)(C)C N1(C(CCOC)=O)CC(CNC(=O)Cc2ccn(CC(C)C)n2)CC1(C)C c1(CCC(=O)NC23C(CN(C(C(CC(C)C)C)=O)C2)CC3)c[nH]c2ccccc12 N1(C(C)C)CCCC(CC(N2CCCCC2CNC(=O)Cc2cncnc2)=O)C1 c1(N2CCC(O)(C(C)NC(=O)CCOC3CC3)CC2)ncnc2c1CCO2 CCS(=O)CC(=O)NC(Cc1ccccc1)CCNC(c1cnc(C(C)O)s1)=O c1(C(N2CC(NC(C(c3ccccc3)C)=O)C(O)C2)=O)cc(Cl)c(F)cc1F C(=O)(CCN(C(c1ccon1)=O)C1CC1)NCCC=CCCC c1(CN2CC(C)N(C(C34CCC(CC3)CC4)=O)CC2)ccc2c(c1)OCO2 c1(C(=O)NCCC(CCNC(C(C=CC)O)=O)C)cc(CC)ccc1Cl c1(N(CC(=O)NCCOC)C)c(F)c(F)c(Br)c(F)c1F C1(CNC(=O)C=Cc2cnc[nH]2)CCCN(C(C2CCCCC2)=O)C1 c1(C(N2CC(CCNC(c3c(C)scn3)=O)OC(C)C2)=O)ncnc2c1CCC2 C1(C(=O)NCC(C)NC(=O)C(C)n2cnnn2)CCNC1=O C1(F)(CNC(CC2(OC)CCC2)=O)CCC(NC(c2cc(C(N)=O)co2)=O)CC1 C1(CC)CC(CC2CN(C(=O)NC(=O)C(C)CCc3ccccc3F)C2)CCO1 C=Cn1nccc1C(=O)NCCC1CCC(NC(c2cc(C3CCC3)on2)=O)C1 C1(c2n(CCOC)nnn2)(NCc2ccccc2OC)CCC(C)SC1 C(=O)(CCC(C)(F)F)N1CCCC(CCNC(COCCC)=O)C1 C(=O)(C(C)(C)CC(F)F)N(CCC1CCN(C(C2(C)CCC(C)C2)=O)CC1)C C1(C(=O)NCC(CC)NC(C2C(C)(CC)C2)=O)CSCCS1 C1(C(C)C)CN(C(c2scnc2Cl)=O)CCN1C(C1CCCN1C)=O c1(C(=O)NCC2C(CC)CCN2C(=O)Cc2cnn(C)c2C)nnc(O)nc1O c1(C(=O)NC2CCCC(NC(C(CC)NC(C)=O)=O)C2)cnc2c(ccn2C)c1 c1(C(=O)NC2CCC(C(=O)N=c3nc[nH]s3)CC2)cccc2nc(Cl)sc12 C(C(C(=O)N(C1CC(N)C1)C)C(C)C)NC(c1cc(COC)no1)=O.OC C12(CNC(CCc3cccc(C)c3)=O)CCCN(C(c3n[nH]cc3C)=O)C1C2 c1(NC(c2ccc(CCC)cc2)=O)cccc(NC(=O)N(C)C)c1C CC1COCC2(CCC2)N1C(=O)Cn1cc(C(F)(F)F)cc(Cl)c1=O N1(C(c2c(C)nc(C)o2)=O)CCCC2(CCCN(Cc3cc(Br)ccc3F)C2)C1 C(=O)(C#CC1CCCCC1)NC(C1(O)CN(C(c2cc(CC)[nH]n2)=O)C1)C c1(C(=O)NC2CCC(NC(CC3C(C)(C)CCO3)=O)CC2)cccc2ncsc12 CCC(C)C(C(=O)NCC1CC(CNC(=O)C=C(C)C)C1)c1ccccc1 CC(CC(=O)N(C)CCn1cc(C(=O)NCC2CN(C3CC3)C2)nn1)C(F)F N1(C(c2c(CCC)cccc2)=O)CCC(NC(=O)C(C)OC(C)=O)C12CCC2 C12(C(=O)NCC(C)CN(C)C(c3csc4nccn34)=O)CCCCN1CCC2 CC(CCC(C)(C)C)C(=O)NCc1ccccc1CN(C)C(C1CCCSS1)=O C(=O)(C(C(=O)NCCCC(=O)NC1(CO)CC(F)C1)OC)OCC c1(N(C(c2ccnc(-c3ncccn3)c2)=O)CC)ccc(Cl)c(-c2cc[nH]n2)c1 c1(OC)ccc(Cl)c(C(=O)N(C2CN(C(C3CCCCC3C)=O)C2)C)c1 N1(C(C2CCC(C)(C)C2)C(=O)NC(CC)(C)C)CCC12CCSCC2 c1(CC)cn2c(C(=O)NCC3(O)CC(NC(=O)C=C(Cl)Cl)C3)cccc2n1 O=C(N=c1[nH]nc(Cl)cc1Br)C1CC(O)CN1Cc1cccnc1Br C1(NC(c2ccc(OC)o2)=O)C=CCN(C(=O)Cc2ccc(C(C)=O)s2)C1 C1(NC(CN(C(=O)CC(C)n2cccn2)C(C)C)=O)CC(=O)NC(=O)C1 N1(C(C)=O)CCCCC1C(N1CCCCC1CCNC(=O)CCn1ccnc1)=O N1(C(CCC)=O)CC2CCN(C(=O)CC3CCC(C)(C)CO3)CC(C2)C1 CC1Cc2cccc(C(N3CC4(C3)CN(C(=O)CCNC(=O)C3CC3)C4)=O)c2O1 C(CC(C(=O)N1CC(CNC(=O)C(C)(F)F)C1)N(C)C)SC Cc1cc(C)c(C(=O)NCC2(C)CCN(C(C3CCCOC3C)=O)CC2)c(O)c1 C1(CC)(NC(c2ccoc2)=O)CCN(C(c2cc(Br)cnc2C2CC2)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NCCC(C)N(C(C(=O)NC(C)C)=O)C c1(N2CCC(C3(C)CC3)C2)cccc(S(=O)(=O)N2CCCOCC2)n1 c1cc(Cl)ccc1Cl.C1(N(C(=O)OCC)C)CCCN(c2nnnn2CC(C)C)C1 Cc1cccc(C=CC(=O)NC23CC2CN(C(c2ccc(C#N)n2C)=O)C3)c1 C1(N(C(=O)CSC2CCOC2=O)CCC)CCN(C(C2(C)CCCS2)=O)CC1 N1(C(C)C)CC(C(=O)N(C(C)CNC(=O)Cc2cccs2)C)CC1=O N1(C(C(CC)C#N)=O)CCCC2CN(C(c3cn(C4COC4)nn3)=O)CC12 N1(C(CC(C)C)=O)C(C(=O)NCc2cccnc2)CC2CCCC12 C1(CN(C)C)CCN(C(C2CCC=CC2NC(c2cscc2F)=O)=O)CC1 O=C(O)C(F)(F)C(c1ccccc1)NC(=O)CC1CCCCO1 c1(CC(N2CCN(C(c3noc(CC)c3C)=O)CC2)=O)ccc2ncsc2c1 N1(C(=O)NCc2c(SCC)cnn2C)CCC23CCC(CC12)C3(C)C c1(C(=O)NC2CC2CNC(C(CC)C(C)O)=O)ccc2oc(C)nc2c1 C=CC1(C(N2CCN(C(C3CCC3)=O)C(CC3CC3)C2)=O)CCCCC1 C(CC(=O)NCCC1CCCC2CC12)(C(C)(C)C)NC(C(C(C)(C)C)=O)=O c1(OC)ccnc(OC)c1C(=O)NCC(O)CNC(c1cc(F)cs1)=O C1(NC(c2nc(C(C)(C)C)oc2)=O)CCN(C(c2ncc(Cl)cc2F)=O)C12CC2 c1(C(=O)NC2CCS(=O)(=O)C2)cccc(OCc2ccccc2)c1Cl C1(C(=O)NC(C2CCCN2c2cc(Cl)ncn2)(C)C)CCc2nnc(O)cc2C1 C1(C(N2CC(C)(NC(c3cccc(CC)c3C)=O)C2)=O)CCc2cnnn2C1 c1(C(N2CCN(C(c3csc(C)c3N)=O)C3C2C3)=O)ccc(S(N)(=O)=O)o1 C1(c2cn(N3CC(NC)CC3=O)nn2)CCN(C(c2ccccc2C)=O)C12CC2 Cc1cc(C)c2nc(NC(c3cc4c(nc3N)CCCC4)=O)cn2c1 N1C(=NCC2COCCO2)N2CCCC(C1CCCCC(C)(C)C)C2 C1(CC(=O)NC(C)C(CO)NC(C2CN(C3CCOCC3)C2)=O)CCCOCC1 c1(CC(=O)NC(C(C)(C)CO)c2ccccc2)cccc(C#N)c1 Cc1nc(C(=O)NCC2C3CN(C(=O)CCOCC(C)(C)C)CC23)nn1C CCC(COC)C(=O)NC(C)CN(C)C(c1c(O)noc1C)=O C1(CNC(C(n2c(C)cc(C)n2)C)=O)CC2CC1CN2C(=O)C=C(Cl)Cl c1(OC)nc(C)ccc1CN1CC(C)CC1C(=O)Nc1cnn(C2CC2)c1 N1(C(C2(F)CCN(C(c3c(C(C)C)occ3)=O)C2)=O)CCOC(C)(C)C1C CC(CN(C(c1cccc(O)c1)C(=O)NC1CCCC1)C)C(C)(C)C C(C)(C)(C#Cc1cn(C2COCC2O)nn1)NC(C=C(C)C(C)C)=O C1(C)(CNC(C2(OC(C)C)CCC2)=O)CCN(C(C2(C)CC2(F)F)=O)C1 CCC(C)(CNC(=O)CC1CCOC1=O)NC(=O)C=C(C)C(C)C Nc1cccc(-c2cn(CCCn3cccnc3=O)nn2)c1.N1(CC)CCOCC1 c1(C(=O)NCCCCNC(c2cccc(CC)c2)=O)cccc2c1OCO2 N1(C(CN(c2ccnc(Cl)n2)C)=O)CCOC(C(=O)NCc2nncn2C)C1 CC1CN(C(=O)C(O)CNC(N)=O)CCC1C(=O)N.C(C(F)(F)F)=C(C)C c1(C(N2CCC(O)(CNC(C=Cc3scc(C)n3)=O)C2)=O)cccc2oncc12 CC1CN(C(=O)CN2CCC(O)CC2)CCC1CNC(c1ncccn1)=O CCCCCC(CCCCC)C(=O)NCCOCCOCCNC(=O)C(C)(O)C(C)C C1(CCN(C(=O)CC2CC(=O)C2)C)CCN(C(C23CCCCC2C3)=O)CC1 CCCCCC(F)C(=O)NCC1(OC)CN(C(=O)C(C(C)C)N(C)C)C1 Cc1cc(CCC(=O)NCCOC2CN(C(=O)C(F)CC3CC3)C2)cc(C)n1 N1(C(CC(=O)OCC)=O)CCCC12CCN(C(c1sc(C(C)C)nc1C)=O)C2 c1(C(N(C2CCCN(C(C(c3cccnc3)C)=O)C2)C)=O)ccc2n[nH]cc2n1 CCC(CC(F)(F)F)C(=O)N1CCN(c2ccc(F)cc2C)CC1 C1(NC(CC2(C)CC2(Cl)Cl)=O)CN(C(=O)CN2CCCCCC2=O)CC1(C)C C1(C(N2CC(C)(NC(c3cocc3C)=O)C2)=O)(NC(C)=O)CCCC1 N1(C(CCOCC)=O)CC2CN(C(C3CCCN3C)=O)CC12 C(=O)(CCCC(=O)C1CC1)N(CCC(C(C)C)NC(=O)CCCCNC(N)=O)C c1(NC(C2(C(=O)N(C3CC3)Cc3cncnc3)CC2)=O)c(Cl)cccc1[N+](=O)[O-] C1(C(=O)NC(c2ccccc2)(C)C)CN(C(C2CCCC3CC23)=O)CCO1 C1(C(=O)NCCCSCC)CCN(C(=O)C2(C#N)CCCOC2)O1 N1(C(c2ccnc(C)n2)=O)CCC(C)C(CNC(=O)C2=CCSC2)C1 Cc1ccc(-c2nc(C(=O)N(CC(C)CNC(c3ccsc3C)=O)C)cs2)cn1 C1(NC(CN2C(C)CC2)=O)CN(C(=O)CCc2ccc(F)nc2)CC1O c1(-c2nccc(C(=O)NCc3cc(Br)no3)c2)ccc(F)c2[nH]ncc12 C(=O)(C1CCc2ccc(C(=O)O)cc21)N1CCC(N(C(=O)C(C)(C)C)C)CC1 c1(C(=O)NCC2(CN(C(C(C(C)OC)O)=O)C)CC2)c[nH]c2cc(F)ccc12 CC1CC2CN(C(C3CC=CCO3)=O)CC2N1C(c1cnc2cccnc2c1)=O CCC(C(=O)NC(C1(NCC2CC2Cl)CC1)=O)C(C)C c1(C(N(CC(O)CNC(c2cnncc2O)=O)C)=O)cc2cccc(Cl)c2[nH]1 c1(OC)c(C(N2CC3CC2C3CNC(=O)C(C)C2CCOC2)=O)ccnc1Cl Cc1cccc2cc(COC(c3cc(C(F)(F)F)cn3C)=O)[nH]c12 N1(C(C2C(CC)C2)=O)CCC(n2cc(Cn3nc(C)cc3C)nn2)CC1 c1(SC(C)C(=O)N(C2CC(NC(C3CC(O)C3)=O)C2)C)ccc(F)cc1 c1(C(=O)NC2C(CNC(CCc3ccc(C)s3)=O)C2)cc(-n2ccnc2)ccn1 CC1CCN(C(C2C3CC(=O)CC23)=O)C1CNC(=O)C(C)(Cl)Cl C(=O)(C1=C(C)N(C)c2ncnn2C1)N(C(C)CNC(=O)CCCCC(N)=O)CC C(=O)(C(C)(C)CNC(=O)CCCc1ncco1)NC(C(=O)NC(CC)C)C c1(C(N(c2ccc(CC)cc2)C)=O)ccc2cnn(C)c2c1 N1(C(c2csc(C(=O)OC)n2)=O)CC(OCC)CC(C)(C)C1 c1(CNC(=O)Nc2c(C)cccc2)cn2ccc(-c3ccnc(O)c3)cc2n1 C1(NC(c2ccc(OC)cc2OC)=O)CCN(C)C2(CC2)C1 C(=O)(CCC(C)(C)C(=O)OC)N1CC(CNC(C(C=CCCC)O)=O)N(C)CC1 C(=O)(C1=CCC(c2ccccc2)C1)N1C(C(=O)OC(C)(C)C)C(C)(C)CC1 C(CC(=O)NCC1(C)CC2CC2C1)(C(F)F)NC(c1c(CC)c[nH]c1)=O CC(O)C(C)CN=c1cc[nH]cc1S(=O)(=O)NC1(COC(C)(C)C)CC1 c1(OC)ccccc1C(=O)NC(C)(C)CCNC(CNC(c1ccsn1)=O)=O S(=O)(=O)(c1ccnc(NC(c2coc(C)c2)=O)c1)N1CCC(SC)CC1 c1(CC(N2C(CCNC(C3C=CCC3)=O)CCC2)=O)cc(F)ccc1Br C1(NC(C2N(Cc3cn(-c4ccn(C)n4)nn3)CCC2)=O)CCN2CCCC2C1 CN1CCC(C(=O)NCC(c2ccccc2)CNC(=O)CC(F)F)CC1 C1(NC(=O)C=Cc2ccoc2)CC2CC1CN2C(c1cnsc1)=O CC1COC(C(N2CC(N(C)C(c3cc(C4CC4)on3)=O)C2)=O)C1 C1(F)(C(=O)NCCNC(=O)NCc2cccc(F)c2)C2CCCC12 O=C1CCCC(CC(=O)NCc2ccccc2CNC(C2CSCCS2)=O)O1 c1(C(N2C(CNC(Cc3ccc(SC)cc3)=O)CC2)=O)cc2cccnc2s1 C12(C(=O)NCC3CC(C(C)C)C3)CCC(CN(C(C3CCOC3)=O)C1)C2 c1(CCC(=O)NC(CC)CNC(=O)C(C)CC2CC2)nc(C)c(C)o1 C1(N(C(=O)Cc2ccoc2)CC)CCN(C(C2CCCCN2S(C)(=O)=O)=O)CC1 N1(C(CN(CCOC)C)=O)CC(NC(c2c(Cl)nn(C)c2Cl)=O)CC(F)C1 C1(CC(N2CCN(C(C#CC(C)(C)C)=O)CC2=O)=O)Cc2ccc(Cl)cc2C1=O N1(C(COC2(C)CCOCC2)=O)CCC(C2CC2)C1CNC(c1cccnn1)=O C(=O)(C(CC)NC(c1ccc(NC(=O)CN2CCCCC2)s1)=O)NCCC c1(C(N(C)CCc2ncnc(Cl)c2CO)=O)ccc([N+](=O)[O-])cc1S(C)(=O)=O O=C(NNc1ccc(Br)cc1)C(CO)c1ccc(Cl)cc1.c1(N)ncc(Br)cc1O C(=O)(CC(COC)NC(C1CN(C)C(=O)N1)=O)Nc1c(CC)nsc1 N1(Cc2ccc(OCC)nc2)CC(C(=O)NC(C)(CO)CO)CC(F)(F)C1 OC1CN(Cc2csc(CCc3ccccc3)n2)C2(CCCC2)C1 c1(C(=O)NCC(CC)(C)Cl)coc2c1CN(C(C1CCC(C#N)CC1)=O)C2 N1(C(C(C(C)(C)O)F)=O)CCCC2(CCC2NC(=O)COCC(F)F)C1 Cc1cn2cc(C(N3CCC4(CCC4NC(=O)C(F)F)CC3)=O)cc(C)c2n1 CC(C)CC(O)C(=O)NCC1(C)CCCN(C(=O)CCc2cscn2)C1 C1(N(C(C(CC)OC)=O)C)CCCN(C(c2ccc(-c3ccccc3)cn2)=O)C1 N1(CCCF)CCC2CCN(c3ccc([N+](=O)[O-])cc3)CC2C1.O=CC=C(Cl)Cl CCCCCCC(=O)NCC(C1(NC(=O)CC2CCOC(C)(C)C2)CCC1)=O C1(C(=O)NC2CCC(NC(C3(CO)CCOCC3)=O)CC2)CN2CCC1CC2 CN1CCC(O)(CNC(C23CCC(N(C)C)(CC2)C3)=O)CC1.C12CC(C1)NC2=O c1(C(N(C2CCCN(C(=O)C(F)(F)C(O)C3CC3)C2)C)=O)cnc2occc2c1 CCC(CC(=O)NCC1CCCC1NC(c1cc(Cl)c(Cl)[nH]1)=O)C(F)F c1(OC)ccc2nccc(C(N3CC(CNC(=O)C(CC)NC(C)=O)C3)=O)c2c1 c1(C(N(CCC(C(C)C)NC(CCC)=O)C)=O)c[nH]c2cccc(C)c12 Cc1nc(C(=O)NCCC(=O)NC2CC23CC(O)C3)sc1C c1(CC)ccc(C(=O)NCC2(NC(=O)C(C)n3ccnc3)CCOCC2)c(C)n1 CC1(C)C(=O)NCCN1C(=O)C1=NOC(C2(O)COC2)C1 C1(CNC(CN2CCC(C)C2)=O)CN(C(=O)CC2=CCCC2)CC(C)(C)C1 CC1CC2(CCC2)CN1C(c1cc(CNC(=O)C(=C2CCCCC2)F)[nH]n1)=O C(=O)(N(CCCO)OC)C1CN(C(C(CC)OC)=O)CC12CC2 C1(C(=O)NC2(c3ccc(F)c(F)c3)CC2)CCN(Cc2ccc(F)cn2)CC1F N(C1CCc2cc(CNC(=O)CSCC)ccc21)C(CNS(CCCC)(=O)=O)=O C1(O)(CNC(C2C(CCC)C2)=O)CCCN(C(=O)C(=CC2CCC(C)CC2)C)C1 Cc1cc(N(C)C)ccc1C(=O)NC1CCN(C(c2cc[nH]c(=N)c2)=O)C2CC12 N1(C(CC(C)(C)C(F)F)=O)CCC2C(CCCN2C(c2cc(O)cc(=O)o2)=O)C1 C(=O)(C(C(C)C)C1CCC1)NCC1C(CNC(CCC=C(C)C)=O)C1 n1(C(C)C)ncc(C(N2CCC(O)(C(C)NC(c3cccnn3)=O)C2)=O)c1F N1(C(CC(C(C)C)C)=O)CCCC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C2 Cc1cc(C(=O)N(CC(C)NC(=O)C(CO)c2ccccc2)C)n[nH]1 C(=O)(C1CCCc2nnn(C)c21)NC1(CC)CCCN(C(=O)CO)C1 c1(NC(C2(c3cc(Cl)cc(Br)c3)CCCC2)=O)c(Cl)ccc(O)c1Cl N1(C(C(C)OC2COC2)=O)CCC(NC(=O)C2=C(Cl)CCOC2)C12CCCC2 Cc1cc(C(=O)NCC2CCC(C(=O)NCC3(C)CCCC3O)CC2)nc(C)n1 C1(C(=O)Nc2c(C(C(=O)OC)C)ccc(Br)c2)CC2CCC(C1)C2F C1(C(=O)NCC(C#C)OC)CCN(C(=O)Cc2cn(C)cn2)C1(C)C c1(N2C3C(NC(C4C(=C)CC4)=O)CC(CC3)C2)nc(Cl)nc(C)c1[N+](=O)[O-] CC(O)(CNC(=O)C(Cc1ccoc1)NC(C1CC2(CC2)C1)=O)CO C1(C(=O)Nc2sccc2CO)CCC12CCCN(C(=O)Cn1nccn1)C2 Cc1ccc(C)c(OCC(N2CCC(NC(C3CCC(=O)N(C4CC4)C3)=O)C2)=O)c1 c1(C(=O)NCCNC(=O)CC2(F)COC2)cncc(-c2ccsc2)c1 c1(CN(C)C(C2CCCCC2)C)cccc(Cc2c(C(=O)OC)ncs2)c1 N1(CCNC(=O)NC2CCCCCC2)CCCOCC12CCCC2 C=CC(CCC)CC(=O)N1CC2CC2(NC(c2cccc(C3(C#N)CC3)c2)=O)C1 C12(CC(=O)NC3(C(=O)OC)CCC3)CCC1CN(C(C1CCC(N(C)C)C1)=O)C2 CCC(CNC(=O)CC1CCCC(C)O1)(CC)NC(=O)CCN1CCCCC1 CCCCC(CCCC)C(=O)NCC(F)CNC(=O)COC(C)CC Cc1cc(C)n2ncc(C(N3CCC(NC(C4(C)CC=CCO4)=O)C3)=O)c2n1 CCCCCC(CC)C(=O)NC(C)CCc1nnnn1-c1ccccc1 C1(C(N(CCCNC(c2c(C(C)C)n[nH]c2)=O)C(C)C)=O)CCCOC1C C1(NC(CSCC=C)=O)CCCN(C(c2sncc2C)=O)C1CC c1(N)cc(CO)ccc1OC.c1(C(=O)C(c2n(C(C(=O)C)CC)nnn2)=O)ccc(Br)cc1C=O.NC c1(C(=O)NC2CC(C(N3CCC(C)(C)C3)=O)OCC2)cc(O)cc(=O)o1 N1(C(=O)OCC)CCCC(NC(=O)CN(CC(C)(C)C)C)C1.C12CCC(CC1)N2 C(=O)(CC(C)CC(=O)NC(c1nocc1C(=O)NC1CC2CCCC2C1)C)OC CC1CC(O)CN(C(c2cccc(C(C)(C)C)n2)C(=O)NC2CC2)C1 c1(OC)cc(C(N2CCC(NC(=O)Cc3c(F)cccc3F)C2C)=O)ccc1C C12(CNC(=O)Cn3nnc(=O)[nH]3)CN(C(c3cnc4n3CCS4)=O)CC1CCO2 N1(C(C(CC=C)OC)=O)CC2CC(O)C1C2NC(=O)Cn1ccc(C2CC2)n1 C1(C(NOCC=C)=O)CCC(C)(C)N(C(=O)CC2CCOCC2)C1 c1(-c2cn(CC3N(C(CCC(=C)Cl)=O)CCC3)nn2)cccc(F)c1Cl c1(C(=O)NCC2(Cn3cc(CCC#N)nn3)CC2)sc2cc(Br)ccc2c1Cl CC1CN(C(=O)CCCC(N)=O)CC(C)C1NC(=O)C(C)n1ccnc1 N1(C(CC2(OC)CN(Cc3nn(C)cc3C)C2)=O)CC2CCC(CC2)C1 N1(C(C(CC#C)C)=O)CCC2C1CCCN2C(=O)Cc1ccon1 c1(C(=O)NOCC2CCCO2)ccc2cccc(F)c2n1 N1(C(c2c(CC)noc2)=O)CC2CC1C2CNC(c1c(C)noc1C(F)(F)F)=O c1(C(N2C(CNC(C3CCc4c[nH]nc4C3)=O)C=CC2)=O)cc2cccnc2[nH]1 C1(C(N2CCC(Cn3cc(C(C(=O)OC)(C)F)nn3)CC2)=O)CCCCC(=O)N1 c1(C(=O)NC2CCC(CC(=O)NCc3onc(CC(C)C)n3)C2)cccnc1O c1(-c2c(OC)cc(C)cc2)ccc2cc(NCc3nocc3C)ncc2c1 C1(NC(C(CC)OC)=O)CCN(C(c2cnn3cc[nH]c(=O)c23)=O)CC12CCC2 CCCC(C)(CC)C(=O)NC1CC(CC(=O)NC2CCN(CCF)C2)C1 C1(C(=O)Nc2n(C)nnn2)CC(F)(F)CN1C(C1CC1c1ccccc1)=O CN1CC(NC(=O)C2=CCC(NC(=O)CCC3CCC(=O)C3)C2)C2(CC2)C1=O c1(C(=O)NCC2CC(NC(c3c(C)nc(C)[nH]3)=O)C2(C)C)ccc2ncnn2c1 c1(C(N2CCC(C)C2CNC(c2cc3cscc3s2)=O)=O)cc2occc2n1C N1(C(Cn2c(C)nnn2)=O)CC(NC(C2CCCCC2(F)F)=O)C2CCCCC12 C1(C2CC2)(C(=O)NCC(C)(CO)CO)CN(C(=O)CN2CCNC2=O)C1 c1(CN(C(c2ccc(Cl)nc2)C(=O)NC)C)cc(Cl)c(O)c(Br)c1 N1(S(CC=C)(=O)=O)CCn2nc(C(=O)Nc3c(C)cccc3C)cc2C1 c1(C(=O)NC(CC)CNC(C2CC(F)(CO)C2)=O)ncncc1Cl C1(C(N(C(C)C2CC2)C2CC2)=O)CN(C(c2coc(C(F)F)c2)=O)CCC1(C)C c1(OC)ccc(OCC(=O)NCCCCN(C(=O)C(C)(C2CC2)OC)C)cc1 CC1(C2CCN(C(=O)C(C3CCN(C(c4cnc(S)nc4)=O)C3)F)C2)CC1 C1(NC(c2nc(C)oc2)=O)CN(C(C2(CNS(N)(=O)=O)CC2)=O)CC1O C1(C(=O)NC(C(C)SC)C)N(C(=O)CCS(C)(=O)=O)CC12CCCC2 N1(C(c2c(C)nccc2)=O)CCC(C)(C)C1CC(=O)NCc1cc(O)ns1 C1(OCC)(OCC(N2CCC(OC)C2)=O)Oc2ccc(OC)cc21.C(C(=O)N)CC Cc1ncc([N+](=O)[O-])n1CC(=O)NCC(C)(C)CNC(C1CCCC1C)=O CCCCC(CC(=O)NCC)NC(=O)C(C)OC(C)(C)C.C(=O)(C(O)COC)N N1(C(C(CCC=C)NC(=O)Cc2csnn2)=O)CCN(C)C(=O)C1C C1(CNC(CCOCC#C)=O)CC(O)C12CCC2.C12CC(CCO1)NC2=O N1(CC(=O)NCC(C2CCCC2)NC(COCCCCC)=O)CCCC1=O Cc1ncccc1C(=O)NCCC(C)(C)CNC(=O)CCCc1nncn1C N1(C(C(CCC)C)=O)C(C)CC2CN(C(=O)CCCF)CC12 N1(C(C(C)N(C)C)=O)CCN(C(=O)CN2C(=O)CN(C)C2=O)CC1C1CC1 Cn1cnc2c(NCC3(CC4CCC4)CC3)nc(N3CCOCC(CO)C3)nc12 N1(C(CCOCCC)=O)CCCC(NC(=O)COC(F)(F)F)C1C C1(O)(CNC(C=Cc2n(C)cnc2)=O)CCCN(C(=O)CC(C)(C)O)CC1 C1(C(=O)NC(c2c(Cl)ccc(F)c2OC)CC)CNCC12CCCCC2 CC1=C(C(=O)NCC2(NC(c3ccc(C(F)(F)F)cc3)=O)CC2)C(=O)OC1(C)C O=C(CC1=CCCC1)NCC1(CNC(=O)C(F)(F)c2ccccc2)CC1(F)F N1(C(CC2C(C)CN(C(=O)C(C)CO)C2)=O)CCN(C)C(C)C1 C#CCC(C(=O)N1CCC(NC(c2ccc(N(C)C)nc2)=O)C1C(C)C)C1CC1 C(N=c1[nH]cnc(N(CC(C)(C)S(C)(=O)=O)C)c1C)C1CC(OC)C12CCC2 c1(C(N(C)CC2COCCN2C(=O)CN2CC3CC3C2)=O)n[nH]c2c1COCC2 Cc1ccc(F)c(C(N2CCC(CNC(=O)C(C)(O)Cc3ccccc3)C2)=O)c1 N1(C(CCN(CC#C)C(C2CCC(C)(CC)O2)=O)=O)CCC(NC(=O)OC)CC1 N1(c2nncc(OC)n2)CC(NC(c2ccc(N(C)C)cc2)=O)CC(C)C1 c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)C(C)(C)CSC)C3)cc1 C1(C(=O)NC(C=C)C2CC2)(NC(C2CCCN2C(=O)OC)=O)CC(F)C1 c1(NC(CC2CCCC(NC(c3n(C=C)ncc3)=O)C2)=O)ccc(C)nc1C c1(C(N2C(CN(C(CSCC=C)=O)CC)CCC2)=O)cc(N)ccc1C N1(C(C=CC(CC)C)=O)CC2CCCC2C1C(=O)NCC(C)(C)F c12ccc(cc1)C(=O)NCC(C)N(C)C(=O)COC2.C1(C(C)SC)CCCCCC1 CC1CN2CCN1CC2C(=O)NC1(CCNC(=O)CC2CCCSC2)CC1 C1(NC(c2ccc(C)s2)=O)CC2CCC(C1C)N2C(=O)C(c1cnn(C)c1)C c1(C(N2C3CN(C(C4CCN(C(C)=O)CC4)=O)C(C3)C2)=O)cccc(C)c1C#N C1(NC(CC2CCC(OC)CC2)=O)CN(C(C2(F)CCOC2)=O)CC12CC2 N1(C(CC=CCC)=O)CCOCC1CC(=O)NC(CO)C(C)(C)C N1(C(c2c(C)csc2)=O)CCCCC(NC(=O)CSC2CCCCO2)C1 N1(C(C2(NC(CC(C)C(F)F)=O)CC(O)C2)=O)C2CCC1CC(F)C2 CCCC(C)C(c1nnnn1CC1CCCO1)Nc1cc(Cl)n(C)n1 n1(CC(=O)N(CCNC(=O)C(O)Cn2cncn2)CC)cnc2c1CCCC2 N1(C(C(C)SC)=O)CC(NC(c2cscc2SC)=O)CC1(C)C C1(CC(=O)NCC(CC)NC(=O)C(C)(C)CSC)SC2=NCCN2C1=O N1(C(C(c2ccccc2)C)=O)CCOCC(C(=O)NC(CO)C2(O)CC2)C1 N1(CC(=O)NC2C(OC)CN(C(CS(CC)(=O)=O)=O)C2)C(=O)NC(C)(C)C1=O N1(C(C2C(C(=O)OC)C2)=O)CC(C2CCCN(C(=O)CCCC3CCCC3)C2)C1 C(CCCC(CO)NC(=O)C(C)C1CCCC1)NC(c1c(CC=C)cccc1)=O N1(C(C(CC)C)=O)CCC2CN(C(c3cc4cc(Cl)ccn4n3)=O)CCC12 N1(C(CC(C)(O)c2ccccc2)=O)CCC2CCN(C(=O)C3=NOCC3)C2C1 N1(C(c2ccnc(OC)n2)=O)C(C(=O)N(CC(C)(C)CO)C)CCC12CC2 C1(NCc2c(CCNC(=O)OC(C)(C)C)ocn2)CCCOC1c1cnn(C)c1 CC(C)CC(F)(F)C(=O)NCCCN(C(=O)Cc1ccc(F)c(F)c1)CCO N1(CCC(=O)NCC(C2CC2)NC(c2c(CC)nns2)=O)C(=O)NC(C)(C)C1=O C=CC1COCC1SC.C123CC(CN1C2=O)C3 N1(C(CCCN(C(c2c(CC)oc(C)c2)=O)C)=O)CCc2ncccc2C1 N1(C(C(c2ccc(Cl)s2)C)=O)C2CCCC1CN(C(C1(C)CC=CCO1)=O)C2 c1(C(=O)NC2CCC(CC(=O)NCCN=[N+]=[N-])C2)cc2ccccc2o1 C(=O)(CCCCC(=O)NCC1(CNC(C2CC(C)(O)C2)=O)CC1)NC C12(C)CN(C(C)(C)C1)C2=O.c1(CNC(c2c(CC)cc[nH]2)=O)cccc(O)c1F CC(CC(=O)NCC1(C(=O)NC2(C)CCCC2O)CCCCC1)CC(C)(C)C Cc1nc(C)n(CC(=O)NCc2ccc(C(=O)N(C)CC3(C)CC3)o2)n1 C(C)(C(=O)N1CC(CC(C)NC(C2C=CCC2)=O)C1)NC(C)=O c1(OC)cc(O)c(OC)cc1OCc1nc(-c2cc(C)cc(C)c2)sc1C N1(C(C2C(=C)C2)=O)CCC(CC=C)(NC(=O)COCc2ccccn2)C1 C1(C)(NC(C2CN(C)C(=O)C2)=O)CCCN(C(=O)Cc2c[nH]nc2O)C1 C1(NC(Cn2c(C)c(Cl)cn2)=O)CC(NC(c2cc(C)n(C)c2C)=O)C12CCC2 C1(N(C(C=C(CCN(C)C)Cl)=O)C)CN(C(c2csc(=N)[nH]2)=O)CC1F C(=O)(C(C)(O)C(C)C)N1CC(CC=C)(NC(=O)C(N2CCSCC2)C)C1 C1(C)(NC(CC2C(CNC(c3c(CC)cccc3)=O)C2)=O)C(C)(C)C1(C)C c1(C(N(CCC)CC2CCCO2)=O)cn2c(n1)CCN(CC1CC=CCC1)CC2 C12(C(=O)NCCC(C)NC(C3CCCN(C(N)=O)C3)=O)COC(CF)(C1)C2 CC1(C)C(NC(C2CCNC2=O)=O)CCN1C(c1cnn(CC(F)F)c1)=O c1(-c2cn(CC3CCCC3NC(CCc3cnn(C)n3)=O)nn2)cncc(N)c1 c1(C(N2CC(NC(=O)CC3CCCCC3)C(CO)CC2)=O)ccc2nncn2c1 c1(C(=O)NC2C(CNC(=O)Cn3nnc(C(F)(F)F)n3)C2)ccnnc1S C1(NC(c2cc(CC)c(CC)o2)=O)CN(C(=O)CCCCNC)CC12CC2.SC c1(OC)ccc(-c2cnc(C(N3CCCC3)=O)nc2)cc1OC(=O)C1CC1 C1(NC(C2ON=C(C)C2)=O)C2CC1CN(C(c1ccccc1C(F)(F)F)=O)C2 C1(NC(c2c(C)nns2)=O)CCN(C(C)C(=O)NCc2ccccn2)CC1C C1(C(=O)NCC(CCOC)NC(c2cc(CO)[nH]n2)=O)CCCC1(C)C CCC(C)C(C)C(=O)NC(c1ccc(F)cc1)CNC(c1ncnc(C)c1C)=O C1(F)(CNC(C(C2CC(F)(F)C2)OC)=O)CCN(C(=O)C=Cc2cc[nH]c2)C1 c1(C(=O)NC2C=CCN(C(=O)C3=CSCS3)C2)cncc(-n2ccnn2)c1 C1(C(=O)NCC2(F)CCOC2)(NC(Cc2c(C)n(C)nc2)=O)CCC(C)(C)C1 C=CC1(C(=O)NC2(C3CCCN3C(c3coc(C(C)C)n3)=O)CC2)CCOCC1 c1(C(N2CC(C)C(NCc3cc(F)c(Cl)cc3O)C2)=O)cccc([N+](=O)[O-])c1F N1(C(C(=O)NCC)C(C)C2CCCC2)CCN2CC(O)CC2C1 C(=O)(CC(C)(C)C(=O)NC(C1CN(C(=O)CCOC(C)C)C1)C)OC N1(C(Cc2cc(C)sc2)=O)CCC2(NC(=O)C=CC3CC3)CCCC12 N1(C(CN(C)CC)=O)CCCC1CNC(=O)C(C)(C)n1cnnn1 c1(N)cc(Br)ccc1C.c1(CCC(C2CCCC2)OC)nnnn1CCCF CCC(CCCC(=O)NC1CC(CSC)C1)NC(=O)C=Cc1cncs1 C(=O)(C(CCSC)NC(c1ccc(OCC)cc1)=O)NC(C(=O)OCC)CC C12(NC(c3nc(C)sc3C)=O)CCCC1CN(C(C1COCCO1)=O)C2 C=CCC(C)(C)CC(=O)NCc1scc(C(=O)NCCC2NC(=O)NC2=O)c1 N1(C(Cc2n(C)nc(CC)c2Cl)=O)CC(C)OC2(CCN(C(=O)C(C)C)C2)C1 C1(c2cc(C)on2)CCCN1N1CCC(C(C)N)C1 CC(C)CCC(F)C(=O)NC(C(=O)NC1CCCC(C2CC2)C1)C1(C)CC1 CN1C2CCCC1CN(C(C1C3CCC(C3)C1NC(c1ccc(F)s1)=O)=O)C2 N1(C(Cc2c(C)occ2)=O)CC(NCCCCCF)CC1C(=O)NC C(=O)(CC(C)CC(C)(C)C)NCC1(F)CCC(NC(C2(COC)CC2)=O)C1 N1(C(C(C)OC)=O)CCC2(CCCN(C(c3nscc3Br)=O)C2)CC1 c1(C(=O)NCC2CC(C)N(C(=O)Cc3cnccn3)C2)coc2c1CCCC2 c1(N(C)C)ccc(NC(N2CC3CC(O)C2C3)=O)cc1F c1(C(C(=O)NC2CC(c3cccc(C(C)(F)F)c3)C2)F)ccc(Cl)cc1F C1(C(N(CC(c2nn[nH]n2)C)C)=O)CC2CCCC2N1C(C1C=CCCC1)=O C#Cc1cc(C(=O)NC2CC23CC(NC(=O)CCc2ccccc2)C3)ccc1Cl S(=O)(=O)(c1cccc(C#N)c1)N1CC(NC(C(C)Cc2ccccc2)=O)C(O)C1 N1(C(c2c(CC)cncc2)=O)CC(N(C(=O)C(=O)NCCOC)C)C(C)(C)C1 C1(CCC)CN(C(C2(C#N)CCCOC2)=O)CCN1C(=O)Cc1ccccc1Cl C(=O)(CC(C)CC(C)C)NCC(CC(=O)NCCCc1ccncc1)OC c1(C(N2C(C(C)NC(C=CC(C)(C)SC)=O)CCC2)=O)cnc(C2CC2)nc1 c1(-c2cc(CNc3nnc(SC(C4CCCO4)C)s3)no2)ccc(F)cc1 c1(C(=O)Nc2nccc(SCC)c2)cc(C(F)(F)F)ccc1O Cc1ccc(O)cc1C(=O)NNC(=O)NCc1cncn1C1CC1 c1(CNC2CC3(CC(NC(=O)CCN4CCCC4)C3)C2)cc2ncccc2o1 Cc1cc(C(=O)NC2CC2NC(c2cncc(Cl)c2)=O)ncc1S(N)(=O)=O Cc1cc(Cl)c(C(C)NCC2CCN(CCO)CC2)cn1 N1(C(C(CC=CCC)C)=O)CCC(C)(C)C(C(=O)NC2(C(N)=O)CCC2)C1 c1(C(=O)NCCC(C)SC)ccc(CNC(=O)C=C(C)C)cc1 Cc1cc(C(N2CC(C(=O)NCc3nc(C)c(C)[nH]3)OC(C)C2)=O)c(C)nn1 N1(C(C2C(C(=O)OCC)C2)=O)CCC2(CC1)CC2(C)NCCS(N)(=O)=O C1(NCc2cccc(OCC)c2)CC2CC(NC(=O)OC(C)(C)C)C2C1 C1(C(N2C3C(NC(C4N(C)CCC4)=O)CC(CC3)C2)=O)CCCC12CCOCC2 c1(C(=O)NCCCCC(C)NC(=O)C(C)n2cccn2)noc2ccc(Cl)cc12 N1(C(C2C(C)=CCS2)=O)CCCC(C(=O)NC2(C)CC2(C)C)C1C CCC(C(=O)N1CCC(N(C(=O)CCCOCC)CC2CC2)CC1)C(C)O CCCC(C)(CC)C(=O)NC1CCCN1CC1(C)CCN(c2ccncn2)CC1 O=C(CC1=CCCCC1)NC1CCC(NCC2(Cc3cccs3)CCOCC2)C1 Cn1cc(NC(=O)CCC2CCN(C(=O)CCn3ccnn3)C2)c(C#N)n1 N1(C(CCC(=C)Cl)=O)CC2(CCN(C(C3CN4CCCN3CC4)=O)CC2)C1 N1(C(C(CCNC(C(C)(C)NC(=O)OC)=O)(C)C)=O)CC2CSCC2C1 c1(C(=O)NC(C)CNC(c2cc(Cn3cc(Cl)cn3)on2)=O)nccc(Cl)c1C C1(C(N(C(C)C2CC2)C)=O)(CNC(C2CCCC(=O)O2)=O)CCCCC1 c1(N(C)Cc2ccc(C)c(C)c2)nc(N2CCCNC(=O)C2)c2c(n1)COC2 c1(C(N(C(CNC(=O)C(C)(C)C(F)F)C2CC2)C)=O)ccc2nc[nH]c2c1 C1(NC(c2c(C(C)(C)C)ncs2)=O)CCC2CCN(C(=O)Cc3cccs3)C12 c1(CC(=O)NC2CCN(c3nc(C4CCCC4)ns3)C2)ccc(F)cn1 C1(NC(C(C)(C)C)=O)CCCCC1CNC(c1ccc(-c2cc(O)ns2)cc1)=O N1(C(C(C2CN(C(CN(CCCC)CC)=O)C2)O)=O)CCCC(OC2CCC2)C1 CCCC(CC(C)C)C(=O)N1CC2(CCN2C(=O)C2=CCCC2)C1 CCC(CC(=O)NC(Cn1cccn1)C(=O)N1CC(OC(=O)N(C)C)C1)OC c1(C(=O)NC23C(CN(C(C=C(C)Cl)=O)C2)C3)sccc1S(C)(=O)=O c1(CNC(c2c(C(N)=O)ccs2)=O)ncccc1CNC(C1(CO)CCC1)=O N1(C(c2nn(CC)nc2Br)C(=O)NCC)Cc2nc(Br)sc2C1 C(C(=O)N=c1cc(-c2cccnc2)[nH][nH]1)(c1cccc(OC)c1)OC c1(C(C(=O)NCC(CNC(COC)=O)C)O)ccc(C(C)C)cc1 C#Cc1cn(C)nc1C(N1CC2CCC2(CC(N2CC3(CC(O)C3)C2)=O)C1)=O Cn1ccc2c(C(=O)NC3CC34CCN(C(C35CCCC3C5)=O)CC4)ncnc12 C1(C(=O)NC2CN(C(C3CC3F)=O)CC2O)COC2(CO)CC1C2.c1ccc(Cl)s1 C1(CC(=O)NC(CCC=C)C2CC2)C2CCC(C2)N1C(C1CC(=C2CC2)C1)=O C(C(CC(F)(F)F)NC(=O)CNC(c1cccnc1)=O)NC(C(CC)SC)=O c1(C(C(=O)NCC2CCN(C(c3cncn3C(C)C)=O)C2)(F)F)cc(Cl)sc1Cl Cc1ccc2c(c1)N(C(=O)CC1(NC(C3CCCN3C=O)=O)CC1)CC2 CCC(CC)CCC(=O)N1CCOC(C(C)NC(C2CN3CCN2CC3)=O)C1 c1(C(=O)NCc2c(C)nn(C)c2C)c(F)cc(Br)cc1Cl Cc1c(NCC2CN(C3CCC3)C2)nc[nH]c1=NCC1(CC2CC2)CCOC1 c1(C(=O)NC2CCC(CNC(=O)CN3CC4CCC3C4)C2)ccc(O)c(F)c1F Cc1ccc(F)cc1CC(N1CC(CNC(c2cccc(Br)c2O)=O)C1)=O Cc1c(C(=O)Nc2cncc(OCC(=O)O)c2)oc2ccccc12 Nc1c(Cl)ccc(F)c1C(N1C2CCC1C(NC(c1cnc[nH]1)=O)C2)=O c1(CC(N2C(CN(C(C(C(C)C)C)=O)C)CCC2)=O)ccc(Br)c(C#N)c1 N1(Cc2scc(C)n2)CCN(C(c2csc(CCP(C)(C)=O)n2)=O)CC1 N1(C(C(C(=O)OC)C)=O)C2CCC1C1CC1(NC(=O)CCc1cccc(C)c1)C2 C1(CC(N2C(CC(=O)NCCOC(C)C)CC2)=O)CC1(C)C C=CCN=C(NCCC(C)(C)CO)NCC1(c2ccccc2)COCCO1 Cc1csc2c(CC(=O)NC3CC4CN(C(c5cnn[nH]5)=O)CC4C3)cccc12 c1(NC(=O)NCC(C(C)c2ccccc2)O)nccn2nc(Br)cc12 N1(C(CCCCOC)=O)C2CCCC1CC(NC(c1cc(C(C)=O)c(C)o1)=O)C2 Cc1ccc(C(CNC(C2CC2(Cl)Cl)=O)NC(c2ccn(CCO)c2C)=O)cc1 c1(C(N2C(CC(NOCC(C)(C)O)=O)CC3(CC3)C2)=O)csc(S(C)(=O)=O)c1 C=CC(F)(F)C(=O)NCC1(F)CN(C(c2cnn(CC3CCCC3)c2)=O)C1 C=CCN(Cc1ccccc1)N1CCC(CCOC)C(F)(F)C1 C(=O)(C(F)(F)C(O)C(C)C)NCC1CC(NC(c2cccc(C(C)=O)c2)=O)C1 c1(CC)nc(C(N2CCCC2C2CCN(C(c3cnsc3)=O)C2)=O)c(N)s1 C1(CNC(CNS(C)(=O)=O)=O)CC2CC1CN2C(C1C=CCC1)=O N1(C(c2sncc2C)C(=O)NC(CC)C)CCCCC1CC(C)C c1(C(=O)OC)ccc(C(=O)NC2(C(=O)O)CCC2)cc1OC c1(CC(N2C(C(=O)NCC3C(CC)C3)CN(C)CC2)=O)c(O)nc(=N)[nH]c1C c1(C(C)(C)C(N2CCN(C(=O)COCP(C)(C)=O)CC2)=O)ccc(C#N)cc1 C1(CNC(c2cscc2Br)CCOC)CCC2(CCC2)O1 c1(C(=O)NCCNC(c2ccc(C#N)[nH]2)=O)cccn2c(Br)cnc12 C1(n2cnnn2)(CC(N2CCC(NC(=O)Cc3ccco3)C2)=O)CCSCC1 Cc1cccc(C(N2CC(NC(C3CC=CCO3)=O)CC(C)C2)=O)c1C C1(CNC(C(C)(C)NC(=O)OC)=O)COCCN1C(c1cnccc1C)=O c1(-n2c(-c3ncccc3N(C)C)nc(CSC)n2)cc(Cl)nc(Cl)c1 c1(C(=O)NCCC(C)NC(c2cccc3ccnn23)=O)ccc(P(C)(C)=O)cn1 c1(C(C)NC(C(COC)NC(=O)C(C)c2cc[nH]n2)=O)c(C)n[nH]c1C C1(CNC(C(COC)(C)C)=O)CC2CCC1N2C(=O)CSc1cccs1 O=S(=O)(c1ccc(SCCOCCO)cc1)N1CCC(C(F)(F)F)C1 C1(C(=O)NCCN(CC(C)O)C(=O)Cc2sc(SC)nc2C)(CC)CCCCO1 N1(C(c2cc(C)n(C)c2)=O)CC2CC(NC(c3nncn3C)=O)C2C1 CC1(O)CCCN(C(C2CCC=CC2NC(C2CCCC(=O)C2)=O)=O)C1 N1(C(C(CC)=CC)=O)CCOC(CCNC(c2cnccc2NC(C)=O)=O)C1 C1(C(N(C(C)CN(C)C(C2(C)CCOCC2)=O)C)=O)CCN(C)C(=O)C1 CC(C(=O)N1CC(O)(CCNC(C23CCC(F)C2CC3)=O)C1)S(C)(=O)=O CS(=O)CCC(O)C(=O)N1CC(O)(CCNC(c2cc(Cl)ccc2N)=O)C1 C1(n2cc(-c3cc(C)ncn3)nn2)CCCC(NC(c2cccc(Cl)c2)=O)CC1 C1(NC(CC=C(C)C)=O)CCN(C(=O)C(C)(C)C(C)C)CC1(C)C Cc1cccc(F)c1CC(N1CC2CC1C2NC(=O)Cn1nnc(=O)[nH]1)=O N(C(=NCCc1ccc(Br)c(F)c1)NCc1ncc[nH]c1=O)CCOCC N1(C(c2cnc3ccnn3c2)C(=O)NC(CC)(C)C)CCCN2CCCC2C1 C1(C(=O)NC(CCC)C(=O)OC)CN(C(=O)NC)CC1(C)C n1(CC)nc(C)c(C(=O)NC(C)CC(C)NC(c2cncc(COC)c2)=O)c1Cl c1(CCN(C(c2cn(-c3ccncc3)nn2)C(=O)NC)C)ccc(S(N)(=O)=O)s1 N1(C(C=C(COC)C)=O)CCCC(CCC(=O)NC(CCO)C2CC2)C1 c1(CNC2CCC(C(=O)NC(C=C)CO)OC2)cc(Br)cc(Br)c1F C(c1cccc(N)c1)=CC(N1CC(OC)(CNC(C2OCCC2C)=O)C1)=O C(=O)(C1Cc2ccc(Cl)cc21)NCc1ccn(CCC)n1 c1(C(N(CCNC(c2ccn(CCC)n2)=O)C2CC2)=O)cc(Cl)c(OC)cc1Cl Cc1c(C(=O)NC(CNC(C2CCCOC2C(C)C)=O)CO)ccc2cncn12 NS(=O)(=O)CCCC(=O)NCC1CC(NC(C2CC3CCC2CC3)=O)C1 CC(CC1CCOCC1)C(C(=O)NC1CCOC1)N(C1CCN(C)CC1)C N1(CC(N2C(CCn3cc(CC)nn3)CC2)=O)CCC2(CC1)CCS2 C#CCC(CC(=O)N(C)CCn1cncn1)NC(=O)C(CCCC)N(C)C C(c1cccnc1)=CC(=O)NCC(N1CCOCC1C1CCCNC1)=O Cc1ccc(NC(=O)C(N2CC(CC(=O)NC3CC3)OC(C)C2)=O)c2[nH]ncc12 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(CCNC(c2cn(C)c(O)n2)=O)CC1C C(CS(=O)(=O)CCN=c1[nH]c(=NCC(C)OC)[nH]c2c(F)cccc12)OC C1(C(N2CCC(C)(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)CC2(CCOCC2)CO1 Cn1cc(-c2ncco2)cn1.N1(CC(=O)N2CC(=O)N3CC(C3)C2)CCOCC1 C=CCC(CNC(c1ncccc1Cl)=O)C(=O)NC(COC)C1(C)CC1 C(=O)(CC(C(F)(F)F)N(C(=O)Cn1ncccc1=O)CC)N1CCCC(C)(CO)C1 Cc1ccc(C)c(C(N2CCC(C)(NC(c3csc(C(F)F)c3)=O)C2)=O)c1N C1(C(=O)NCC(=C)Br)CN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1(C)C N1(C(CC(CNC(CC(=O)NCC#C)=O)OC)=O)Cc2ccccc2C1 C1(NC(CC(C)C)=O)CN(C(c2nc(C(C)(C)C)cc(O)n2)=O)CCC1C Cn1cc(CCNC(=O)C#CCNC(=O)CSCCC#N)cn1 N1(C(Cc2cccc(C)c2)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1C Cc1ncc(Br)c(N2CCC(NC(=O)C(C)n3ccnc3)C(O)C2)n1 N1(C(C2(OC)CCC2)=O)CC2(CCOCC2)C1c1cn(Cc2cc(Cl)no2)nn1 CCCCCC(CC)C(=O)NCC1CC(F)CN1C(c1ccn2c1CCCC2)=O C1(C)(C(=O)NC2CCC(CCNC(CC3CN(C)C3)=O)C2)CC2CC2C1 C(=O)(C(CC(C)C)ONC(C1CCC1)=O)N(c1ccsn1)CC.C1(N)COCCC1CO c1(OC)c(O)cc(C(=O)NCC2(NC(=O)CSCC(N)=O)CC2)cc1C#N C(=O)(C(F)C(F)(F)F)N1C(CNC(c2c(OC)noc2C2CC2)=O)CC1 c1(C(N(C2CCCC2)CCCNC(C2OCC(C)C2)=O)=O)cnc2occc2c1 N1(CC2(c3nnnn3C3CC3)CC(CC)NCC2)CCC2(CCCNC2)CC1 Cc1c(C(=O)NCC2CCN(C(=O)Cc3ccc(F)cn3)C(C)C2)cccc1F c1(CN(CCCNC(c2cccc(OC)c2)=O)C(C2C(C#C)C2)=O)cc(N)ccn1 C1(C(C(=O)NCC2CCOC2)N(CC(F)F)C(C)C)CCCC(C)C1 C(=O)(C1=CCCC1)N1CC(C)(O)C1.O=C(CCOC1COC1)NCCO C1(C(=O)Nc2ccnn2Cc2ccccn2)CC2(CCN1)CC2 c1(C(C(N2CC(N(C(CCOCC(C)C)=O)C)C2)=O)O)ccc(F)c(F)c1 c1(CC(=O)NCC2CC(CNC(c3c(C)cno3)=O)C2)ccccc1C(F)(F)F c1(C(C(=O)NCC2CN(C(c3cnc(C)[nH]3)=O)CC2O)C)nc(F)ccc1Cl N(C(=NCc1cccc(-c2nccn2C)c1)NCC(C)(C)C(=O)C1CC1)C(C)C C1(C(=O)NCC2(CCNC(C(C(C)C)O)=O)CC2)CCc2ncnn2C1 n1(CC(=O)NC2CN(C(C(C(C)C)NC(N)=O)=O)CC2O)ncc2ncccc12 N1(C(C(C=C)O)=O)CCC(O)(C(C)NC(=O)Cc2cccc(OC)c2)C1 c1(OC)cc(F)ccc1C(=O)NCC1CN(C(=O)Cc2ccc(Cl)s2)CCCO1 N1(C(C(C2CCCCC2)OC)=O)CC2CC(NC(C3(C)CC3)=O)CC(C2)C1 c1(C(=O)NC(C(=O)N(CC)CC2(O)CCC2)CCC2CC2)ccc(C)c(O)n1 C(=O)(C1=C(C#N)CCC1)NCC1CCN(C(C(CC(C)C)C)=O)CC1C C1(CNC(C(C)N(C)C)=O)CN(C(=O)CCc2cccnc2F)CC(C)(C)O1 c1(C(N(C)CC2N(C(C(COC)(F)F)=O)CCC2)=O)c(F)c(F)cc(F)c1F c1(C(=O)NC2CN(C(c3c[nH]nc3F)=O)CCC2O)cc2cncn2c(O)n1 c1(CCNC(C2(CCCOC)CCCC2)=O)cc(Cl)sc1Cl C1(NC(C2N(C(C)=O)CCC2)=O)C2CC(NC(c3csc(Cl)c3)=O)CC12 C12(NC(C3(COC)CCC3)=O)COC(CNC(C3CC3(Cl)Cl)=O)(C1)C2 C(C(C(=O)N1CCc2nn[nH]c21)C(C)C)NC(COCc1c(C)cccc1)=O c1(-c2ccc(C(C)C)cc2)nc(CC2CCCCC2)n(C2CCc3ccccc32)n1 c1(CCC(N2CCC(O)(CNC(C3CCC(C)CC3)=O)C2)=O)cc2ccccc2[nH]1 C1(C(=O)NCC(CC)NC(c2cnc[nH]c2=N)=O)CC(c2ccccc2)=NO1 c1(NC(c2n(CCSC)nnn2)c2csc(C)n2)ccc2c(c1)C(=O)N(C)C2 NS(=O)(=O)c1cc(C(=O)NCCCNC(C2(CC3CC3)CCCC2)=O)cs1 CC(c1ccccc1Cl)=CC(=O)NCCN1CCN(c2nc(C#N)c(Cl)s2)CC1 CN=c1[nH]nc(CC(=O)NC(C)C(C)NC(c2csc(C)c2C)=O)s1 C(c1ccc2c(c1)OCO2)=CC(=O)NCCNC(C1(C)C(C)CCCC1)=O C=CCC(CC)C(=O)NCCc1cc(C(=O)NCCSCS(C)(=O)=O)no1 N1(C(=O)CCC2CCC2)CCC(C2CCCN(CCc3ccc(F)cc3)C2)CC1 C1(C(C)NC(c2n(C(C)C)ncc2)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1 C1(CCCNC(=O)CCNC(c2cccs2)=O)CCCN1C(c1ccsc1)=O C1(NC(c2c(C)nc[nH]2)=O)COC2(C1)CN(C(=O)C(=Cc1cccnc1)F)C2 N1(C(CCCCCNC(C)=O)=O)CCC2(CCN(C(=O)Cc3cnsc3)CC2)C1 c1(C(N2CC(NC(C(CC)(C#N)CC)=O)C(C)C2)=O)cncc2ccc(F)cc12 c1(CNC(C2CCC(O)C2)=O)nocc1C(=O)N(CC(F)F)CCO Cc1ccccc1CCNC(=O)C=CC1CCCN1C(=O)C(C)O n1(CC(=O)NC2CC(CNC(=O)C(F)(F)C3CC3)C2)ncc2cccnc12 N1(C(C)=O)CCC(F)C(NC(c2cnc(N3CCOCC3)nc2)=O)C1 c1(NC)c(C(=O)NC2CN(C(=O)C3=C(C#N)CCC3)CC2C)cccc1[N+](=O)[O-] c1(CNC(=O)NCc2ncc(C(C)(F)F)s2)cccnc1-n1cccn1 C(C1(CC(=O)N(C)C)CCOc2ccccc21)Nc1ncc(OC)cn1 CC1CC(NC(C2(N(C)C)CCOCC2)=O)CN(C(C2(C3CCC3)CC2)=O)C1 C(C(=O)NC1CCOCC1)(C(C1CCOC1)OC)N(CCOC)CC CCC(CC)(C(=O)NC(c1ccc(F)cc1)CNC(=O)CSC1CCCC1)OC C(=O)(C(C(C)C)NC(C1CCC1C#N)=O)NCc1c(C)nns1 c1(C(=O)NCC2(CCNC(C(C(CC)O)C)=O)CC2)cc2cc(C)ccc2cn1 CCC(C)C(C(C(=O)NCc1ccco1)N1C2CCCC1COC2)OC Cc1cc2c(cc1C)N(C(C1(C)CC3(CCC3)C1)=O)CC2 C(=O)(C1=CCCOCC1)NCC(CNC(C(C)CF)=O)(C)C c1(C(=O)NC2CN(C(CC3(C)CCCCC3)=O)C2)cc2nc(F)ccc2o1 CN1C(=O)CCC1C(=O)NCC(c1cccc(Cl)c1)NC(C1CC12CC2)=O c1(C(=O)NCCNC(C(=O)NCC)=O)cccc(NC(C2CC3(CC3)C2)=O)c1 Cc1nc(C)n(CCCC(=O)NC2CC(O)(CNC(=O)CC3(C)OCCO3)C2)n1 c1(C(N2CCCC(F)(CNC(C(COC)(F)F)=O)C2)=O)cc(=O)n2nccc2[nH]1 C1(CCN(C(C=C(CCC)C)=O)C)CCCCN1C(c1cc(COC)ccn1)=O N1(C(C(C)=CC)=O)CC(C)CN(C(=O)Cc2c(F)cccc2Br)CC1C c1(ONC(=O)NCC(C)CNS(C)(=O)=O)ccccc1CCP(C)(C)=O C(=O)(CCC(C)S(C)(=O)=O)N1C(CN(C(C(CC=C)(F)F)=O)C)CCCC1 CC1CC(C)(C(=O)NC2CCN(C(=O)COCCN(C)C)CC2CO)CCO1 c1(C(N2CCN(C(c3nccc(CC)c3)=O)C(C)C2)=O)c(C)cc(C)cc1O N1(C(C2N(C)C(=O)CC2)=O)CCN(C(=O)C(=O)NCC2CC2)CC1CC1CC1 N1(C(C2N(C(CCC)=O)CCC2)=O)CC(NC(C2CCCN2C)=O)CC(F)(F)C1 C12(NC(c3cc(SC)oc3C)=O)CCCN(C(=O)Cn3c(C)csc3=O)CC1C2 C1(OC)CCCC1NC(C1(CC2CC2)CCC1)=O.C12CCCN1C2=O Cc1ccccc1OCC(=O)NC1(CNC(C2(c3ccncc3)CC2)=O)CCC1 C12(CNC(C3CC(C(C)C)C3)=O)CCC1CN(C(=O)CCc1cccc(O)c1)C2 Cc1conc1CNC(C1CCCC1CNC(C1CCC1C(F)(F)F)=O)=O c1(N(C)C)ncc(C(=O)NCC2CN(C(c3ccnn3CF)=O)CCO2)cc1Cl N=c1cc[nH]cc1CC1CN(C(C2CCN(c3ccccc3)CC2)=O)C1 CC1(NC(C2CC(=O)CCO2)=O)CCN(C(C2C3CCCC23)=O)CC1 C(C(CC(F)(F)F)NC(C12CCC1C2)=O)NC(c1cncc(C(N)=O)c1)=O C(=O)(CC(=O)NCC(O)CCNC(=O)C(O)C1CN(C(C)=O)C1)N(C)C.C(C)(C)C CCC(Cc1ccccc1)CC(=O)NC1CC(NC(C2(F)CC3(CCC3)C2)=O)C1 c1(C(COC(=O)CN(C)C(c2ccn(C)n2)=O)OC)ccccc1C c1(C(N(C)Cc2nc(N3CC(c4ccccc4)C3)sn2)=O)cc(O)nn1C C(=O)(CCC(CF)CF)NC(c1ccccc1)C(=O)NCC1(O)CCC(C)C1 C1(CNC(Cc2cccc(SC)c2)=O)CN(C(=O)CCC2CC2)C2CCCC2O1 c1(C(N2C(CNC(c3ccc([N+](=O)[O-])[nH]3)=O)CCC2)=O)cc(Cl)cc(Cl)c1O N1(C(C2OCC(C)C2)=O)CC2CCCN(C(c3ccc(-c4ccco4)o3)=O)C2C1 CC1(CNC(C2(C#N)CC2)=O)CCC(NC(c2csc(C(N)=O)n2)=O)C1 c1(OC)cc(OC)c(F)c(CNC2CC(CC(=O)NC3CC3(F)F)C2)c1F CC12CC1(C)CN(N(Cc1cccc(C(N)=O)c1)COC(F)F)CC2(F)F c1(CCNC(=O)Nc2cscc2-c2ccccc2)ccc(O)nn1 c1(N2CCN(C(c3ncc(OC(C)C)nc3)=O)CC2)nnccc1C#N C1(C(=O)Nc2ccc(C(=O)OC)cc2C)CC2(C1)NCCN1CCCC21 C(=O)(C(C)CC(C)C)N(CCCC(N1C(C)(COC)C=CC1)=O)C CCCCCCC(C)(CCC)C(=O)NC(C)CNC(c1ccn2ccnc2n1)=O C1(COC)CCN(C(C2(CNC(=O)C=CC3CC3)CC(C)(C)C2)=O)CC1 C1(C)(C(N2CCC(C(C)NC(CC(CC)O)=O)C2)=O)CCCCCC1 c1(C(N2CCCC(CC=C)(NC(C3CCC(F)C3)=O)C2)=O)c(C)cc(=O)oc1C CCC(C)C(O)C(=O)NCC1CC(NC(c2ccc(CO)nc2)=O)C1 C1(CCNC(c2c[nH]c(Br)c2)=O)CCCCN1C(c1ccc(CO)nc1)=O C(=O)(C1=COCCO1)N1CCC(CNC(CC(C)C)=O)C1 C#Cc1cc(F)c(C(=O)NCC2CC(C)(C)CN2C(c2csc(C)c2)=O)cc1F C1(CC(C)NC(CC=C)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C)cc1 c1(CC2(O)CCN(CC(c3ccccc3)OC)CC2)c(F)cccc1Cl C(=O)(C(C)(C)C(=O)NCC1CC(O)CN1C(C1CC1C(=O)OC)=O)NC C1(NC(C2ON=C(C)C2)=O)CC12CCN(C(=O)C1=COCCO1)CC2 C(=O)(CC(C)S(=O)(=O)NC(=O)CN1CC2N(C(=O)C3CC3)CCC2C1)OC CC1CC(C#N)(C(N2CCOC(CC(=O)NCCCc3nncs3)C2)=O)C1 CC1(O)CCN(C(C2(NC(C34CCCC3CCC4)=O)CC2)=O)CC1O C1(C(=O)NCC(=O)NCC(=O)N(CC(CCC)C)C)CSCC(=O)N1 Cc1ccc(C(C)NS(=O)(=O)C2CC2c2cccc(F)c2)c(C)c1 Cc1nccc(Cl)c1C(=O)NCC1C(C)CCCN1C(=O)C1=NOCC1 C1(CNC(c2cn(CC=C)nn2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 c1(CNC(C)=O)ccc(C(=O)N(C2CC(NC(C3CC=CC3)=O)C2)C)cc1 Cn1cc(Cl)cc1C(=O)NCC1(C(=O)NCC2CC(F)(F)C2)CC1 C1(NC(C)=O)CCN(C(=O)Cn2nnnc2C(C)C)CC12CCC2 C(=O)(C1=CCN(C(=O)CC2CCCC2)CC1)N(C1COC(C)(C)C1)C c1(C(=O)NCCN(CCC)C(C2CC=CCC2)=O)ccncc1-c1ccccc1 N1(C(c2c(C)cc(CC)o2)=O)CC(C(=O)NCCC(=O)OC)CCC1C CC(C)CC(F)C(=O)NCC1C=CC(NC(=O)CCc2cn[nH]c2)C1 CC(C)(O)C(F)(F)C(=O)N1CCC(C(C)C(N2Cc3cccnc3C2)=O)CC1 N1(C(CC2(C(=C)F)CCC2)=O)CCc2[nH]nc(C(=O)NCCc3nccs3)c2C1 c1(NC(C2(C(C)(C)C)CCC(N)(C(C)C)C2)=O)cccc(N=S(C)(C)=O)c1 C(=O)(CC(C)CC(C)(C)C)NCC#CC(N1CCCC(C)(CCC)C1)=O c1(N(CCCNC(S(CC)(=O)=O)=O)C)ccc(C(F)(F)C(F)(F)F)cc1C c1(N(C)CC2(F)CC2)nc(=NCc2ccoc2)[nH]c2c1CSC2 C1(CC(=O)NCCCCCSC)CN(C(c2c(C)n[nH]c2C)=O)CCC1C C1(NC(c2cc(COC)no2)=O)CCOCC1NC(C1CC(n2cccn2)C1)=O CC1CC(CCNC(=O)C=C2CCC2)CCN1C(=O)CC(=O)NC1CC1 N1(C(c2c(C)ccc(O)c2)=O)CCCC(O)(CNC(=O)COCC(F)F)CC1 C(CC(F)F)(C(=O)NCCc1ccns1)NC(C1CCN(C)CC1)=O c1(-n2cc(C(=O)NC3CNCC3C3CC3)nn2)cccc(C#CC2CC2)c1 C(=O)(C1SCCc2ccccc21)N1CC(C)C(NC(C2(C)CCOCC2)=O)CC1 CC(C(=O)NCc1ocnc1C(=O)NC(c1ccnn1C)CO)C(F)F N1(C(c2c(C)cco2)=O)CCC=CC1C(N1CCC(OC2CC2)CC1)=O C#Cc1cc(C(=O)N(C)CC2(O)CN(C(C3CCC3C)=O)C2)cc(Br)c1 N1(Cc2ncn(C)n2)CC2CCN(C(c3cc4cc(Br)ccc4[nH]3)=O)CC2C1 C1(CN(C(CCC)=O)C)CC(F)CN1C(=O)C(C)SCCN(c1ccccc1)C C1(CC(=O)NC(CCN(C(c2c(CCC)nns2)=O)C)C)CCC(=O)N1C CCC(CCCC(=O)N1CCCC1C(C)(C)O)NC(c1cccc(=O)o1)=O CCC(C)CCCCC(=O)NCC(CC(C)C)NC(c1ccc2occc2n1)=O CC1Cc2c(Cl)c(Br)cc(F)c2CN1N1CCCC1c1ncccn1 N1(C(n2nccn2)C)CCC(CC(=O)O)CC12CC2 N1(C(C2CCN(C(C(CC=C)C)=O)C2C(C)C)=O)CCC12CCC(C)CC2 C1(C(N(C)Cc2ccncc2)=O)CC2(CCC2)CN1C(=O)Cc1cnn(CCl)c1 CC1=C(C)CC(C(=O)NC2CC(CCC(=O)NC34CC3CN(C)C4)C2)CC1 N1(C(c2ncc(C)cc2C)=O)CCC(NC(=O)C(F)(F)C(C)(C)O)C(C)(C)C1 CC(C)C(N=c1nc2[nH][nH]cc-2c(O)n1)C(C)NC(c1cc2cccnc2[nH]1)=O N1(C(C2(COC(C)C)CC2)=O)CCC2CN(C(C3CCC=CO3)=O)CC2CC1 C1(C)(C(N2CCC(C)(CNC(c3c(CC)c[nH]n3)=O)C2)=O)CCCNC1=O C1(OC)(CNC(C2CC(Cl)(Cl)C2)=O)CCN(C(=O)CCC2C(=O)NN=C2C)CC1 C(=O)(C1=CCC(NC(c2ccccc2F)=O)C1)N(C)CC1(O)CCCC1 C(CC(C)(C)C(=O)NCc1cccc(O)c1)NC(c1c(C)ccnc1)=O c1(C(=O)NCC(CC(C)C)NC(C(CC)(C)C(N)=O)=O)cc(C#N)c(F)cc1F CC(C)CCCC(C)C(=O)NCC1COCCN1C(c1ccnn1C)=O C1(C(=O)NC(CN(C(C2(CC#C)CC2)=O)C)C)CN(C)CCO1 C1(CNC(c2cc(C)[nH]n2)=O)CN(C(=O)CCCN2C(=O)CNC2=O)CCO1 C1(C)(C(N(CC(=O)NC(c2scnc2C)C)CCC)=O)CCC2CC2C1 CCC(C(=O)NCC(C)CN(C)C(c1ncccc1COC)=O)C(C)O N1(C(C(=O)N(C(CCC)C)CCOC)=O)CCc2c(O)cccc2C1 C(=O)(CC(C)C(C)(C)C)NCC(CNC(C(C(CC)C)OC)=O)OC C1(CNC(C(C)SC)=O)CCC2(CC1)CCN(C(C1CCC3(CC1)N=N3)=O)CC2 c1(C(=O)NCCC2CCCN(C(c3ccno3)=O)C2)cnc2c(F)cccn12 Cc1ccc(C(=O)NC2(C3CN(C(C4CC(O)C4)=O)C3)CC2)c(F)c1Cl N1(C(C(CCC=C)NC(=O)Cc2cccs2)=O)CC2C(=O)NC(=O)C2C1 c1(C(=O)OC2CCCC(OC)C2)cccn(C(C)(C)C)c1=O c1(CC(C)C(=O)N2CCC(N(CCO)CC3CN(C)C3)C2)ccc(F)cc1 C(=O)(CCCCCF)NC1C(OC)CN(C(=O)CCCC2CCOCC2)C1 N1(CC(CC)Cc2ccc(Cl)cc2)CCC(F)CC1(C)C CC1CCC(CC(=O)NCCn2cc(C(=O)N(C3CCC3)C3CC3)cn2)C1 c1(C(N(CCCNC(=O)Cc2nccn2C)C(C)C)=O)sc(F)cc1Cl c1(CC)nc(C)[nH]c1C(=O)OC(C)(C)C.C1(O)(CNC(=O)O)CC2CCC12 CCC(C)C(C)C(=O)NCc1cc(C(=O)NCC2(C)CCCCC2)ccn1 C12(C(=O)NCC3CN(C(N)=O)C3)CCC(CN(C(c3cncs3)=O)C1)C2 c1(CS(=O)(=O)NC(c2ccc(OC)c(F)c2)C(=O)OCC)ccc(F)c(C)c1 C(=O)(C(F)(F)C(O)CC)OCC(C1CCOC1)OC C1(NC(C(C)CF)=O)CCCN(C(=O)CCOCC2CC2)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N(CC(C)NC(=O)Cc1cc2ccccc2o1)C N1(C(=O)CCCC2CCC2)CCC(F)(F)C(CNC(C2(F)CCCCCC2)=O)C1 N1(C(C2(C)CC(C)C2)=O)CC2(COC(CNC(=O)COCC3CCOCC3)C2)C1 N1(CCN(C(C(C2CC(C(C)C)C2)OCC)=O)C)CCCCC1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2CCC(NC(=O)CCC(=O)N(C)C)(C2)C1 C1(OCCOC)C2CC1N(C(=O)O)C2.C1(C(=O)OC(C)(C)C)(CO)CC(C)(C)C1 C#Cc1ccc(CC(N2CCC(C(=O)Nc3cccc(F)c3)C2C)=O)cc1 CC(CC(=O)N1CC2(CC(CNC(c3cc4c(o3)CCCC4)=O)C2)C1)P(C)(C)=O C1(NC(CSC)=O)CN(C(=O)Cc2nncn2C(C)C)CC1C C1(C(=O)NCCN(C(C(CN(C)C)(F)F)=O)C)OCCOC12CCC2 CN1CCN(C(c2ccn(C)c(=O)c2)=O)CC1=O.c12cn(nn1)C1(CC1)OC2 N1(C(Cc2ccc(SCC)cc2)=O)CC2CN(C(C3CCC(=O)O3)=O)CC2C1 c1(C=O)cn(C)nc1-c1ccncc1.CC(CCN(C1CC1Br)C)NC C(=O)(C(CCC1CC1)NC(c1cc(CCO)on1)=O)NCC(CC)n1cccn1 Cc1ncc(C)c(N2CCC(NC(C3CN4CCN3CC4)=O)C(O)C2)n1 C1(CC(=O)N(C2CC3CCC2CC3)C)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O N1(Cc2ccc(SC)s2)CC2CCC1CN2C(c1cc(Br)cnc1C)=O N1(C(c2c(C(C)C)ocn2)=O)CC2(C1)CN(C(C1C3CCCC13)=O)CCO2 C(=O)(C(CNC(=O)C(F)CC1CCOC1)N(C)C)N(CC(=O)OC)CC1CC1 C(=O)(C(C)(C)C1CCN(C(=O)C(O)CF)C1)NCCCOC=C c1(C(=O)NC2C(C)N(C(c3csc(O)n3)=O)CCC2)ccc2c(c1)CCCC2 c1(C(N2CCC(C(C)NC(=O)C(C)(C)F)C2)=O)cc(C(F)(F)F)cc(F)c1 C1(CNC(CCC=C)=O)COCCN(C(c2ccc(C)c(CO)c2)=O)C1 N#Cc1nc(Br)cnc1NC(C1CCCN(C(c2cncc3sccc23)=O)C1)=O Cc1ccc(CN=c2[nH]c(-c3cncc(OC(C)C)n3)cs2)c(SC)c1 CC1CN(C(C2(N(C)C)CCC2)=O)CCC1NC(c1c(C(F)(F)F)ncn1O)=O C1(CN(C(C(C(CC)C)N(C)C)=O)C)CCC2(CCNCC2)CC1 C(=O)(C(CC(C)C)NC(=O)OC)N(CC(CNC(c1noc(CC)c1C)=O)C)C Cn1c(NC(=O)C(C)(C)c2nccs2)cc2sccc12 c1(C(N2CCC(CNC(C=CCCC)=O)C23CC3)=O)cc2cc(Cl)ccc2s1 N1(C(CC2(CNC(C3C(CCC)CCC3)=O)CC2)=O)CCC(C2(O)CC2)CC1 c1(NC(C)=O)cccc(F)c1C(=O)NC1CN(C(=O)C2CC2)CC1F C1(OCC)CCCN(C(=O)C(CSCC)NC(=O)CCC(C)N(C)C)C1 CC#CCCC(=O)N1CCCC(NC(C2(C)CC2(C)C)=O)C1 C1(NC(C(C)S(N)(=O)=O)=O)COC2(C1)CN(C(=O)C#CC1(C)COC1)C2 N1(C(C2=CC(C)CC2)=O)C2CCC1CN(C(=O)CCCN1CCCC1)C2 C1(CCNC(c2cn[nH]c2)=O)CN(C(c2cn(CC(F)(F)F)cn2)=O)CCCO1 c1(C(C(=O)NC(CC)(C)C)N(C)CC2CCOC2)csc(C(C)(C)C)n1 Cc1cc(NC(=O)C(F)(CNC(=O)C(C)(C)C(C)C)C(C)C)c(C)cc1F c1(C(=O)NCCN(CCOC)C(c2cc(COC)sn2)=O)n[nH]cc1C1CC1 c1(OC)nccc(Br)c1C(=O)NC1C=CC(NC(C2CCCOC2)=O)C1 N1(C(C(C2CCC(C(=O)O)CC2)F)=O)CCC2C(C1)C2(F)F c1(C(=O)NC2(CC(=O)NCC(C(C)O)O)CCCCC2)ccn(C)c(=O)c1 c1(C(=O)NC2CCC(NC(c3ccon3)=O)C2)cc(C(F)(F)F)ncn1 C12(CNC(C(C)=CC3CC3)=O)CCCC1N(C(=O)CC(O)C1CC1)CCC2 c1(CC(=O)NC2C(CNC(CN(C)CC)=O)CC2)c[nH]c2cc(Cl)ccc12 C1(C(C)C)CN(C(=O)CC2CCSCC2)CCN1C(C1CCOC1)=O CC1=C(C(=O)N2CCC(C)(NC(C3CCCC(C(N)=O)C3)=O)C2)C(C)(C)CCC1 c1(-c2n(C)ncn2)ccccc1CNC1CCC1NC(C1CCC(O)CC1)=O c1(C(=O)NCC2CC(NC(C(CC#C)CC#C)=O)C2)cnc2ccc(C)cn12 c1(C(=O)NCC2(CC(=O)NC)CCOCC2)cc(Cl)c(Br)cn1 CN(C(=NCC1CCC1)NCC1(c2ccccc2F)CCC1)C1CCC1 C=CCCCC(=O)NCC(C)NC(c1ncoc1-c1ccccc1F)=O c1(OC)cc(C(N2CCN(Cc3cnc(Cl)cn3)C3CC23)=O)cc(O)c1O C(N=c1nc2c(cnn2C)c(NCC2(COC)CCCCC2)[nH]1)C1N(CC)CCC1 C12(NC(=O)CSc3nc[nH]n3)CC(CC(=O)NC3CN(C(C)=O)C3)(C1)C2 C1(N(C)C(c2ccc(C#N)s2)=O)CCCN(C(=O)CCNc2cncnc2)CC1 N1(C(CCN(CCC)C)=O)CCN(C(=O)CC2CCN(C)C2)CC(O)C1 C1(NC(c2c(N)non2)=O)CC12CC(NC(C1(n3ccnn3)CC1)=O)C2 N1(C(c2cc(CC)nc(O)c2)=O)CC2(COC(CNC(C3(F)CC3)=O)C2)C1 Cn1c(CCC(N2CCCC2(C)C(C)(C)C)=O)nnc1S O=C1OC2CCC1CN(C(C1CCC(C(F)(F)F)CC1)C(=O)N1CCCC1)C2 N1(C(C(CCC)OCC)=O)CCC2(CC1)OCCC2NC(c1cnccc1Cl)=O c1(OC)cc(C)c(C(=O)NCC2(NC(=O)CC(C)CF)CCCC2)cn1 C1(C(C)C(N2CCC(n3ccnc3)C2)=O)CCN(C(C2CC2(F)Cl)=O)CC1 N1(C(c2c(C)nsc2)=O)CCC2(C1)CN(C(=O)CCC1CC1(C)C)C2 c1(C(=O)NCCN(C2CCCC2)C(Cc2c(C)cco2)=O)cncc(Cl)n1 N1(C(C#CC(=O)N(C)C)=O)CCCC(O)(CNC(c2ccc(O)nc2Cl)=O)CC1 N1(C(c2cc(OC)nc(Cl)c2)=O)CCN(C(=O)CC(C)N(C)C)C2CCC12 C1(CC(=O)N(CC(C)NC(CCc2onc(C(C)C)n2)=O)C)CCCC1(F)F C(=O)(C1CCCc2nccn21)NC(CNC(C1=NOC(C)(C)C1)=O)(C)CC1CC1 N(S(=O)(=O)N1CCCC1C)CCCC.c12ccc(cc1F)[nH]2 N1(C(c2ccc3c(c2)COC3)=O)CCC2C(CCCN2C(=O)Cc2ccon2)C1 Cc1cccc(C)c1CN1CCCC(NC(=O)C(C)Cc2c(C)n[nH]c2C)C1 C1(C(=O)NCCCN(c2ccc(Cl)cn2)C(C)C)CC2(C1)CC(F)(F)C2 C(=O)(CCCC(=O)NCC1CCN(C(=O)C(C)OCCC(C)C)CC1)NCCC C1(CNC(c2nc(COC)sc2)=O)CC2(CC2)CN1C(=O)C(C)n1cccc1 CC1SCCCC1C(=O)NC1(C)CC(C(=O)NCCOCCN(C)C)C1 C(C1CCCC1)=CC(=O)NCC1C=CCN1C(c1csc(CC(F)(F)F)n1)=O CCS(=O)CC(=O)NCC1CC(CNC(c2[nH]ccc2-c2ccccc2)=O)C1 C1(C(=O)NC(C)C#N)COC2(CCN(C(c3cc(Br)cn4ccnc34)=O)CC2)C1 N12CCCC1CCNC(=O)C2=O.C(=O)(C(O)CC1CCCC1)NC1CCC1CF CC(C)(O)C(F)C(=O)NCC1CCCC(NC(=O)CC2OCCCO2)C1 c1(OC)cnccc1C(=O)NCC(C1CC1)N(C(=O)C(F)(F)c1csc(=N)[nH]1)C C(C(C)(C)CC(=O)Nc1cncnc1C)NC(c1oc(CC)c(C)c1)=O C1(C(C)NC(C2CN(C(C)=O)C2)=O)CN(C(=O)CC(C)(C)O)CCO1 c1(C(=O)NC2CC(CNC(CN(CCC)C)=O)C2)c(F)ccc(F)c1F N1(C(c2cc(C)c(C)o2)=O)CC2CC1CN2C(=O)C(C)c1cc[nH]n1 S(=O)(=O)(c1ccc2oc(O)nc2c1)N1CCC(F)(C(N2CC(O)C2)=O)CC1 c1(C(=O)Nc2ccccc2OC)nccnc1CC.c1(C(=O)NC)ccco1 c1(C(=O)NCCN(CCOC)C(c2cccc(C(C)(F)F)n2)=O)cc[nH]c(=N)c1 CCCCC(O)C(=O)NCC1CC2(CC2)CN1C(C1CCCN(CC)C1)=O N1(C(c2nc(CC)oc2)=O)CCOC2(CCCN(C(c3c(C)ncn3O)=O)C2)C1 c1(CC(=O)NC2CN(C(CC3CC(=C)C3)=O)C3C2C3)ccc2c(cnn2C)c1 C(C(C)C(F)C(=O)NC1CCOC1(C)C)NC(c1cnc(C(C)C)o1)=O c1(SC)nc(N2CC3(CC3)CC2CNC(c2c(Cl)nsc2Cl)=O)cc(O)n1 CCS(=O)(=O)CC(=O)OCc1c(C(=O)NC2CCN(C)CC2)cccc1 c1(CC(=O)NCC2(OC)CN(C(c3cncc(C)c3)=O)C2)ccccc1C(C)C C(=O)(C1CCc2snnc21)NC1CCCC(NC(C(C)(C)n2ccnn2)=O)C1 N1(C(c2cnn(C)c2Cl)C)CCC(n2cc(C(O)C(C)(C)C)nn2)C(F)(F)C1 C1(C(N2C(CCC(=O)NC3C(CC=C)CCC3)CCC2)=O)CC=C(C)CC1 C(N=c1nc2ncn(C)c2c[nH]1)C1CC(C)N(C(=O)C(c2ccccc2)F)C1 N1(C(CC2=CCN(C(N3C(C)CCCC3C)=O)CC2)=O)CCC2(CC1)CNC2=O C#CC1CCCN(C(=O)C(C)(C2CC2)N(C)C(c2ccn(CC)c2C)=O)CC1 c1(C(=O)NC(CC(C)NC(=O)CSCCC#N)C)noc2ccccc12 C1(CNC(=O)CCC2CCCCO2)CCN(C(=O)C(O)C2CCC2)CC1 C1(C(=O)NCCN(CCC)C(c2cc(CC)nnc2C)=O)CCn2ccnc2C1 c1(CNC(CC2(O)CN(C(CC3CC(OCC)C3)=O)C2)=O)ccncc1CC C(=O)(C(O)CC(N)=O)NCCCN(CCCNC(COCCC)=O)C C(=O)(C(C)CC(F)(F)F)N1CCOCC(NC(CCC2CC(OC)C2)=O)C1 S(=O)(=O)(c1cc(C(=O)NC(c2cn3ccccc3n2)C(=O)O)ccc1C)NC C(C(C)(C(C)C)NC(=O)C(=O)NCC(c1ocnc1C1CC1)=O)OC c1(C(N2CC(CNC(c3ccccc3C(F)F)=O)C2)=O)c[nH]c(=O)cn1 C1(CNC(CC2(C)CCCCC2)=O)CC2(CC2)CN1C(C1CCCC(F)(F)C1)=O C1(C)(C(=O)OC)CC(CC(N2CCC(CNC(=O)C(C)Cc3cnco3)C2)=O)C1 N(C1CCc2ccc(Cl)nc21)C(C(C)NCc1nc[nH]n1)=O C(=O)(C(CC)C(C)(C)CC)NCC(CC)NC(c1ccnc2c1ncn2C)=O C1(CCNC(CCc2onc(CC)n2)=O)CN(C(=O)C(F)=CC2CC2)CCO1 c1(C(=O)NC2CN(C(C3(Cl)CC3)=O)CC2C2CC2)cc(=O)n2ccsc2n1 Cc1nc(C(=O)NCCC(O)CNC(=O)C=CC2CCC2)cc(O)n1 N1(CC(=O)NCC(CO)NC(c2sccc2F)=O)CSCC1=O c1(C(N2C(CCC(=O)NCCCn3ccnn3)CCC2)=O)cc(=O)cc[nH]1 C(C)(C)(C(=O)NCCC1CC(NC(=O)Cc2csc(C(F)(F)F)c2)C1)C1C(C)C1 N1(C(COC(CC)(C)C)=O)CC(C)CN(C(=O)CCCc2ncco2)CC1C C12(NC(C(C)NC(C)=O)=O)CCCN(C(C3CC(=O)N(C)C(=O)C3)=O)CC1C2 c1(C(C)C)ncc(C(=O)N(CC(C)N(C(=O)CCn2ncn(C)c2=O)C)C)n1C C1(CCC)(NC(c2nc(O)sc2C)=O)CCNCC1 N1(c2snc(COC)n2)CC2CC1CCC2NC(C1CCc2nncn2C1)=O N1(c2nc(-c3c(C)sc(Br)c3)on2)CC(C)c2ccccc21 Cc1cc(C(=O)NCCC(C)NC(=O)Cc2ccco2)on1 C12(CNC(=O)Cc3csnn3)CCC1CCN2C(c1cccnn1)=O N1(C(c2cc(C)on2)=O)C2CCC1CC(F)(CNC(c1cnc(O)o1)=O)C2 CCCC(CC)CCC(=O)NCC1(CNC(C2C(C)C2C)=O)CC1 CC(C)(C)CC(O)C(=O)N1CC(C2CC2)(C(N2CCS(=O)C2)=O)C1 CC1CN(C(C23CC(C)(CN2C(=O)CC(C)C(C)(C)C)C3)=O)Cc2c[nH]nc21 c1(CC(=O)NC2C(C)N(C(C3CC3F)=O)CC2)cc2ccccc2cc1O c1(C(N2C3CC(NC(C=C4CCN(C)C4)=O)C(C3)C2)=O)ccc(Cl)c(Cl)c1O N1(C(c2cccc(C)n2)=O)CCC2(CC1)CN(C(C1(F)CC1C)=O)CC(C)O2 Cc1n[nH]c(C)c1CCNC(=O)CC1CSCN1C(=O)CCCC1CCC1 CCS(=O)(=O)CCNC(=O)C=CC(C)C.C(=O)(CC(C)(C)C)N(C)C(C)=O N1(C(C(C)(C)OC(C)=O)=O)CCC(CO)(CNC(=O)C(C)C(F)F)C1 N1(C(C2N(C)CCOC2)=O)CC2CC(Nc3ccncn3)CC1C2 N1(C(CCSCCC)=O)CCC(C)(CNC(=O)C(C2CCC2)OCC)C1 C1(CNC(C(CO)N(C)C)=O)CC(C(=O)NOCc2ccc(F)cc2)=NO1 N1(C(C(CC)=CC)=O)CC(C)CN(C(=O)C(C)(C)OC)CC1C N1(C(C(=CC2CCCC2)C)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C(C(C)C)C1 C1(NC(Cn2c(C)cc(C(F)F)n2)=O)CC2CC1N(C(C1C(C)C1C)=O)C2 C1(C(N2CCN(C(c3c(C)cns3)=O)CC(CO)C2)=O)COc2ccccc2O1 C1(CC)(CNC(C2CCCC2OCC)=O)CCCN1C(=O)C(CO)N(C)C N1(C(C(C)(O)C2CC2)=O)Cc2ccc(CNC(c3ccn(C(F)F)n3)=O)cc2C1 C(=O)(C(CO)N(C)C)NC1(C(=O)NC(c2ccon2)C)CC1 c1(C(N2CCC(N(C)C(=O)OC(C)(C)C)C2)=O)cncc2nc(O)[nH]c12 CC12CC(NC(=O)CC3C=CCC3)(C1)C1(CN(C(C3CCCCC3O)=O)C1)O2 O=S(=O)(c1cncc(Br)c1Cl)NC(c1cncc(Br)c1)c1nnnn1C1CC1 CCCC(C(=O)N1CC(CNC(=O)CCCNC(N)=O)(OCC)C1)NC(C)=O Cc1ccc2cc(C(=O)N(CC(O)CN(C)C(C3CC4CC3C4)=O)C)ccc2c1 C(=O)(C1=CCSC1)N(CC(CC)NC(=O)Cn1ccnn1)C C(=O)(CCCC(=O)NCc1ncoc1C1CCN1C(=O)NC1CCCCC1)OC O=C1CSc2ncc(C(=O)NC3CC3CNC(C3(Cl)CC3(F)F)=O)cc2N1 C(CC(C(C)(C)C)NC(=O)COCC(F)F)N(C(=O)Cc1cncs1)C c1(C(C)(C)C)ccc(N)c(C(=O)NC2CCC2CNC(=O)C(N)=O)c1 c1(NC(N2CCC(c3ccc(=N)[nH]c3)C2)=O)cc(O)nc2ncccc12 Cc1cc(C(=O)NC2(CO)CCCN(C(c3snnc3C)=O)C2)cc(Cl)c1 c1(C(=O)NC2CCN(C(C3(N(C)C)CC3)=O)C2)cc(O)ncc1Br c1(C(N2CCC(N(C(C(COC)C)=O)C)C2)=O)cccc2cncn12 CC(C(O)C(F)F)NC(c1cnn(CCNC(=O)CCc2cnn[nH]2)c1)=O N1(C(CC=CCC)=O)CCCN(C(=O)CCNC(=O)CC(C)C)CC1CC Cc1ncc(Cl)c(C(N2CC(NC(c3cc[nH]c3)=O)CCC2C)=O)n1 C=CC(CC)CC(=O)NC(CC(=O)Nc1cnc(O)cc1C)C1CC1 c1(OCCN(C)C)ccc(NC(=O)N(C2CCC2)CCNS(N)(=O)=O)cc1 C(CC(C)(C)CC(=O)N1CC(C2(NC(=O)C=Cc3ncc[nH]3)CC2)C1)OC c1(C(=O)NC2CC(N(C(C3(CC)CC3)=O)C)C2)cc2cccc(Cl)c2s1 n1(CC)ncc2cc(C(=O)NCCC(C)CCNC(=O)Cc3ccco3)cnc12 Cn1ncc(CC(N2CCC(OCCNC(c3cnns3)=O)C2)=O)n1 c1(C(=O)NCC2CC(NC(=O)COc3ccc(F)cc3)C2)ccccc1[N+](=O)[O-] c1(C(N2CC(CC)C(NC(=O)C(C)(F)F)CC2)=O)ccn2c1CSCC2 C1(N(C(C)C2CC2)C(=O)OC(C)(C)C)CCN(C(=O)C(N)=O)CC1 c1(C(=O)NCCC2C(CC)C2)c(CNC(c2ncc(F)cn2)=O)cnn1C N1(C(C2(SC)CC2)=O)CCC(NC(C2CC(=O)NC(C)C2)=O)C(O)C1 C1(NC(CN(C)C2CC2)=O)CCN(C(=O)Cc2nc[nH]n2)CC1c1ccccc1 N1(C(=O)NCC(C2CCCC2)C)CCC(c2nc(=O)o[nH]2)CC1 n1(CC(=O)NC(C)CN(C)C(c2c[nH]nc2[N+](=O)[O-])=O)sc2ccccc2c1=O C1(C(C)C)CN(C(c2c[nH]cc2C(C)(C)C)=O)CC1NC(=O)CN(C1CCC1)C Cn1ccn2ncc(C(N3CC4(CC(NC(c5cscn5)=O)CO4)C3)=O)c12 C1(NC(c2ccc(OC)nc2)=O)CN(C(=O)Cn2cnnc2)CC12CCOCC2 C1(c2c(C)ocn2)CC2CC1CC2c1nc(C(=O)OC(C)(C)C)no1 c1(C(=O)NCC)cc(C(N2CCC(OC)C2)C(=O)NCC2CCOC2)on1 N1(C(=O)Cc2ccccc2C(F)(F)F)CC2CC1CN2Cc1ccncc1Br C1(C)(NC(C(CC(C)C)N(C(CCOC)=O)C)=O)CC(C)(C)OC1=O C12(OC)CCC(C1)N(CC(N1CCCC1C1CCCOC1)=O)C2 C(=O)(CC1CC(=O)c2ccccc21)NCC(C)NC(=O)CC1CCCCCC1 c1(-c2cn(C(CNC(c3cccc(CC=CC)n3)=O)C)nn2)cccc(C)c1F c1(N(c2n(C)nnn2)CC2CC2)cccc(Cl)c1 C(C(CN=c1[nH]c(N(CCC#N)C)nc2c1COCC2)SC)OC Cc1cc(C(=O)NCC2(O)CC(NC(=O)C(F)Cc3ccccc3)C2)no1 c1(C(=O)NC2CC(C)(NC(CC(C)(C)OC)=O)C2)[nH]cc2c1CCS2(=O)=O c1cnc2ccccc2c1.C1(C(F)(F)F)(CNC(=O)NC(C)(C)C=CCl)CC=CCO1 c1(C(=O)NCC2C(C)CN(C(=O)C(C)(C)CO)C2)nccc2ncncc12 C(=O)(C1CCCc2ccccc21)N1CCC2(C(NC(c3cnco3)=O)C2)CC1 n1(C(C(N2CCC3C(NC(CC(C)C)=O)C32)=O)C)c(=O)oc2ccccc12 C(=O)(CCCC(F)(F)F)N1C(C)CC(CNC(C2COC(=O)N2C)=O)C1 C(=O)(CCCN=[N+]=[N-])N1CC(CC(=O)N(CC(C)SC)C)OCC1 c1(CN(CCC(C)CO)C2CCCC2)cccc(Cl)c1F O=C1NC2CN(C(C3CC(O)CN3C(C3CCCOCC3)=O)=O)CC2O1 C12(CNC(c3cnc(OC)nc3)=O)CCC(CC1)N2C(C1CC(C(C)(C)C)C1)=O N1(C(c2c(C)c[nH]c2)=O)CCC2(C=C(C(=O)NCC(C)(O)CC(C)C)C2)C1 Cc1cccc2c1CC(C(=O)NCC1CCCCN1C(=O)CN(S(C)(=O)=O)C)N2 O=S1(=O)CC2CN(Cc3ccc(S(=O)(=O)NCCCO)s3)CC2C1 c1(C(=O)NC(C)CCNC(=O)CCCC2CC2C)nccnc1N CC(CC(=O)NC(C)(C)C(c1ccccc1)n1cc(-c2ccnn2C)nn1)N(C)C c1(Cn2c(C3CON3)nnn2)ccc(OC)cc1.c1(COC)ccsc1OC N1(c2nc(C)nc(C#N)c2)CC2CCCC(NC(C3(C4CC4)CCCO3)=O)C2C1 c12cnccc1NC(CC)CNC2=O.c1(CC(=O)OC(=O)C2CC2)ccccc1 N1(C(CCN(CCCCC)CC)=O)CC=C(CNC(=O)CN(C)CC)CC1 c1(C(=O)NC2C3CCN(C(C4CC5(CC5)CO4)=O)C23)cc(Cl)c(Cl)c(Cl)c1 CCC(C(=O)N1CCN(C(=O)CC2CCCCCC2)CC1CO)C(C)(F)F C(CCCC(=O)NC1(C2CCCN2C(=O)CCC2CCCO2)CC1)N(C)C N1(C(CC=C(C)C)=O)CC2(C1)CN(C(c1cccc(Cl)c1C(F)(F)F)=O)C2 CC1(C(N2CCC2C(=O)NCC2=CCCOC2)=O)CCNC1=O N1(C(C(C)N2CCCC2)=O)CCC(c2cn(CC3CC4CC4C3)nn2)CC1 c1(NCC2(CNC(C3CN(CCO)CCO3)=O)CC2)cc2n(n1)CCC2 c1(C(=O)NCCOCC)ccc2c(c1)CCN(Cc1ccsc1Cl)C2 c1(C(=O)NCC(O)C2CC2)cccc(OCCNC(C2(C3CC3)CC2)=O)c1 N1(C(CCCSC)=O)CC2C3CCC(C2C1)N(C(c1cc(C)n(C)c1)=O)C3 c1(C(=O)NCC(C)N(C(CN2C(C)CC2)=O)C)cc(Br)c(C(C)=O)s1 c1(C(N2C(CN(C(C(CC#C)C)=O)C3CC3)CCC2)=O)nc(CC)ncc1Cl c1(OC)ccnc(C(N2CC(N(C(=O)C(F)=CC3CC3)C)C2)=O)c1 O=C(C1Cc2ccccc21)N1CCCC(CCNC(C23CCC(CC2)C3)=O)C1 c1(OCC(=O)NCC(C)NC(=O)CCNC(C2CCC2)=O)c(F)c(F)cc(F)c1F c1(C(N2CCC(O)(CNC(=O)CCC(F)F)C2)=O)cc2ccc(F)cc2[nH]1 N1(C(CCOc2ccn(C)n2)=O)CCCC(NC(c2ccncc2F)=O)CC1 N1(C(C2CC3(CC3)C2)=O)CCCC(F)CC1.CC1(C)C2C1C(=O)N2 C=C(C)C1OCCCC1C(=O)NCCCCC1CN(C(C2CC=CC2)=O)C1 CC(C)C(F)C(=O)N(C)CCN(C(=O)CCc1ccc(OC(C)C)cc1)C c1(NC(C2(COC)CN(C(=O)COCCN(C)C)C2)=O)nn(C(C)(C)C)cc1Cl C=CCC(CC(F)F)NC(=O)CC1CCCN(C(=O)Cn2cc(CO)nn2)C1 CC1CN(C(=O)CC2OCCO2)CCC1CNC(C1CC(C(F)(F)F)C1)=O C1(C(=O)NCc2cc(C)ns2)CC(C)CN(C(C2CC(=O)NC(=O)C2)=O)C1 c1(C2(C(=O)NCC(C)(C3CC3)NC(CC(CCC)O)=O)CC2)cc(F)cc(C#N)c1 c1(C(N(CC(C)N(C(CCCc2ncc(C)o2)=O)C)C)=O)cc2ncccn2n1 N1(C(C2(C=C)CCCC2)=O)CC(C(=O)Nc2cnn3ccccc23)C2(CCC2)C1 C12CC13CCN(CC3)CC(=O)N2.Cc1ccc(N2CCN(C=O)CC2)c(I)n1 C(=O)(C(C)CC(F)(F)F)NCC(=CC(N1C2CC(OC)C2CC1)=O)C c1(CC(N2C(CC(=O)N(c3ccccc3)CC)CCC2)=O)ccc(F)c(Cl)c1F N1(C(C2(SCC)CC2)=O)CCC(C)C(NC(=O)C(C)=O)C1 c1(CNC(CC(C=C)(C)C)=O)cccc2c1CCN(C(C1CCC(F)C1)=O)C2 c1(C(=O)NCC(CNC(=O)C2=CCCS2)O)nnc(O)c2ccccc12 C(=O)(CC(C)NC(c1c[nH]nc1CNC(c1cc(C)[nH]n1)=O)=O)NC C#CC1(NC(C2CCC=CC2NC(=O)CN2CC3CC3C2)=O)CC2CCCC12 CCC(CC)C(F)C(=O)N(CC(O)CNC(=O)CC(CC)C1CCC1)C c1(C(=O)NCC(CO)NC(=O)CCNC(C2CCCO2)=O)ccc2nccn2n1 C1(CNC(C=CCC)=O)(CF)CCN(C(=O)CCSc2ccccn2)C1 N1(C(c2ccn(CC)n2)=O)CCC(C2CC2)(NC(c2cn(CCO)nn2)=O)C1 c1(COC(C)(C)C)cccc(S(=N)(=O)C(F)F)c1 c1(OCCN(C)C(C2CC3CCC2CC3)=O)cccc(C(F)(F)F)c1F c1(C(N2CCC(N(C(CCC=C=C)=O)CCO)C2)=O)cnc2c(cnn2C)c1 Cc1c(O)ccc(C(=O)NC(CNC(=O)C(CC2CC2)CC2CC2)CO)c1C Nc1c(Cl)cc(NC(C2CN(Cc3csc(Br)c3)CCS2)=O)cc1Cl CON(C(=O)C=C1CC1C1(c2cc3ccccc3o2)CCCC1)C(C)C c1(C(=O)NC2(C)CCN(C(C3CCC3C(F)(F)F)=O)C2)cccc2c[nH]nc12 N1(c2c(C)cncn2)CCC(O)(C(=O)NC(C(C)C)c2nc[nH]n2)CC1 N1(C(C(C)OCCOC(C)C=CC(=O)O)=O)CC=CC1C(N)=O C1(c2n(CCCSC)nnn2)(NCCCCCCC(C)C)CC2OCCCC12 c1(CNC(c2n(CCC(C)C)nnn2)C2CC3CC3C2)cnc(C(C)(C)C)nc1 C1(NC(c2cc(C)oc2)=O)C(C)CCN(C(c2ccn(CC#N)n2)=O)C1C CC1(C(N2CCC(OCCNC(C3CCCCNC3)=O)C2)=O)CCC2CC2C1 C(CC1=CCN(C(=O)C2CC2)CC1)NC(C1(N(C)C)CC(c2c(C)cco2)C1)=O c1(NC(C(CC)C(C)O)=O)ccc2c(c1)CCCC2NC(=O)OC(C)(C)C N1(C(c2n(CC)ccn2)=O)CCCN(C(C2CC2CC(C)C)=O)C(C(C)C)C1 C(CC)(CC)(CCNC(c1cc(OC)ccc1F)=O)NC(COCCC=C)=O c1(C(=O)NCC(CCCC)NC(=O)CCOC(C)C)[nH]cc2c1CCC2 N1(C(=O)Nc2c(Br)cc(C)c(C)n2)CC2CC1CS(=O)(=O)C2 CCC(C(=O)NCCN(C(=O)COc1ccccc1Br)C)C(C)(C)CC c1(N(C(=O)CCNC(=O)C(c2cncnc2)C)C)cccc(C(N)=O)c1 C(C(CC(C)C)C(=O)NCC(N1CCCC1)=O)NC(C(C=C)C)=O Cc1ccn(C(=O)NCCCOCC(C)(C)C)n1.c12ccc(o1)C(=O)NCCO2 C=CCC(CC(F)F)C(=O)NC1C(C)CN(C(c2cnc(O)c(F)c2)=O)CC1C CC(CNC(=O)C=Cc1ccoc1)CC(=O)NCC(C)(C)F C(=O)(C(CN=[N+]=[N-])NC(=O)Cn1cncn1)N(CC(N1CCCC1)C)C C(=O)(CC(F)(F)C(F)F)N1CC(CNC(c2scc(C)c2)=O)C(C)C1 S(=O)(=O)(c1cccc(=NCCCCCC(F)(F)F)[nH]1)NCC(C(C)O)(C)C C#CC1CN(c2nc(-c3ccccn3)nc(C)c2Br)CCN1C C(=O)(C1OCCn2ccnc21)NC12CN(C(C3CCCC(=O)N3)=O)C(CC1)CC2 c1(CC)ccc(C(N2CC(O)CC2CNC(=O)C(n2cnc(C#N)n2)C)=O)cn1 CC1(C)CC(NC(=O)CC2CCCOC2)CCN(C(=O)C=CCN2CCCC2)C1 c1(OCC(=O)NC2CC(CNC(C3(C)CC3(Cl)Cl)=O)C2)cc(Cl)cc(Cl)c1 c1(C(=O)NC(COC)C(=O)N2CCCC2c2ccc(Cl)cc2)cc(F)cc(F)c1 N1(C(c2c(C(=O)O)c(Br)ccc2)=O)CCC2(CC1)CC(c1ccc(Cl)cc1)C2 c1(C(=O)NCC(CC=C)NC(=O)C=CC=CC)c(C)cc(C)cc1N C1(OC)(CNC(=O)COC2CC2)CCN(C(c2cccc(C(C)(C)C)c2)=O)CC1 Cc1cnc(C(=O)NC(CC2CCC2)C(=O)NC(c2ccccc2O)C)cn1 N1(C(c2c(Cl)ccc(C#N)c2)=O)CCC2CN(C(=O)CSC(F)(F)F)CC2C1 c1(C(c2cn(CCN(C3CCOC3)C)nn2)C(=O)O)ccc(F)cc1 Cc1ccc(O)nc1CNC(=O)CCCC(C)NC(=O)C(F)(F)F C(=O)(C(CC(F)F)NC(c1ccc(C2CCCO2)[nH]1)=O)NCC(C)N(C)C C(=O)(CC(C)(C)CC(F)F)NC1CCN(C(c2c(C(C)C)ncnc2)=O)CC1O Cc1nn(CC(N2CCC(NC(C3CC3(C)C(F)F)=O)C2C)=O)c(C)c1C N1(C(C(C)OC)=O)CCCC(C)(C(=O)NC(Cc2ccco2)CO)C1 C(CCCCCNC(=O)CCn1c(C)csc1=O)NC(CSc1ncc(C)o1)=O c1(CC(=O)NC2C(C)N(C(c3cnn[nH]3)=O)CC2)ccc(Br)c(F)c1 c1(C(=O)OC)cc(CCCCCN(C(=O)C(F)C2CCOC2)C2CCCC2)on1 c1(C(N2CCCCC(CNC(C3CCC(O)C3)=O)C2)=O)ccc2c(n1)NCCO2 N1(C(COCCOCC#C)=O)CCCCC(CNC(c2cnc(S)nc2)=O)C1 C1(NC(C(C)OCC(C)C)=O)CCN(C(c2n[nH]cc2F)=O)C12CCC2 N1(C(=O)CN2CCC(CO)CC2)CCCC2CN(C(=O)CC3CCCOC3)CC12 C(C(C)C(=O)N(Oc1ccccc1)C(C)CC)OC C(=O)(CC(F)(F)CC(=O)NC1CN(C(c2c(C)n[nH]c2C)=O)CC1C)OC CC1=C(C(=O)NC2CCC(CNC(c3cc(O)ccc3O)=O)C2)SCCO1 N1(C(C(C)OC)=O)C2CCCC1CN(C(C1CCN(c3cnccn3)CC1)=O)C2 C(=O)(CC(C)C(C)C(C)C)NC1C2CN(C(c3cc(CC)no3)=O)C1C2 C1(C(N(C(CNC(Cc2cccc(SC)c2)=O)C)C)=O)CCOC2(CCCC2)C1 CCCC(C)CC(=O)NC1(CC(=O)Nc2cc(CO)cc(F)c2)CC1 N1(C(CCCN(C)C)=O)CCCCCC(Nc2ncc3ccnc-3[nH]2)C1 c1(OC)ccc2[nH]c(C)c(C(=O)NC(C)(CSc3ccc(F)cc3)C(=O)O)c2c1 C1(C(C)C)CCN(C(=O)CC(CNC(C2CC(=O)N(C)C2)=O)C2CCC2)CC1 c1(OC)cnccc1-c1ccc(NC(=O)N(C)OC)cc1 c12ccc(nc1)S(=O)(=O)C(=O)NCC(OC)CNC2=O.C1(CC)(CO)CCCC1 N1(C(C2(C)CC2Br)=O)CCC2(CC(NC(=O)COc3ccccc3F)C2)C1 C1(C(=O)NC(CNC(CCc2onc(CC)n2)=O)(C)C2CC2)CC2(CCCO2)C1 C1(CC)(NC(C2CCC(C)(C)C2)=O)CCCN(C(=O)CCCc2ccc(C)s2)C1 C12CN(CC1C)C(=O)NCC2.C1(COC)(OC(C)(C)C)CCC1 C(CCC(C)C)(C(=O)N1CCCN(C)CC1C)NC(C1(SC)CC1)=O C(=O)(C(C)CC(F)(F)F)N1C(CNC(c2cc(C)sn2)=O)CC(C(C)C)CC1 N1(C(C2(OC)CC2)=O)CCC(O)(CN(C)C(C2CC(NS(C)(=O)=O)C2)=O)C1 Cc1sc(Br)nc1C(=O)NC1CCCC1CNC(=O)C(C)CC1CC1 c1(NC(CC#C)COC)ccc(C2CC2)cc1 C(CCCC(=O)N(C(C)CCNC(=O)CC1(CO)CCOCC1)C)OCC Cc1ccc2c(C(=O)NCC3CN(C(=O)C(C)C)CCO3)cnn2c1C N1(C(CCC(=O)OC)=O)CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC1C2 CC(C)(C)C(CNC(c1cnncc1O)=O)C(=O)NCC1(C)CC2CCC1C2 C1(NC(C)=O)C2CC(NC(=O)C(C3(O)CCCC3)F)CC12 C(=O)(C(F)(F)F)NC1CCN(C(CSCC(=O)Nc2cc(Cl)cs2)=O)C1 C(CC(C)CC)(C(=O)Nc1cnn(CC)c1C)NC(C(CC=C)CC)=O N1(C(Cc2c(C)cccn2)=O)CC(CNC(=O)C(F)(F)C2CCCC2)C(C)(C)C1 c1(C(N2C3C(NC(=O)CC4CC=CCC4)CC(C3)C2)=O)c[nH]c2ccc(F)cc12 c1(CN(C(=O)CC2(C)CC2(F)Cl)C)cnn2c1CN(C(=O)CC1(O)CCC1)CC2 CC12CCOC(C(=O)NC(Cc3cnc[nH]3)C(=O)NC3(CO)CC3)(C1)C2 N=c1[nH]c(Cl)cc(=NC2CCCC3CN(C(c4cc(Cl)c(Cl)[nH]4)=O)CC23)[nH]1 c1(OCC)cc(NC2(CNC(=O)CC3CCCC4(CC4)C3)COC2)nc(C)n1 CON=C(C(=O)N1CCC(C)(NC(=O)CCCN(C)N=O)C1)c1ccco1 N1(C(C=CSC)=O)CC2CC(NC(=O)Cc3ccc(F)cc3)C1C2 c1(CNC(CCC(=C)C)c2nnnn2CSc2ccccc2)cccc(Cl)c1C N1(C(CCC)=O)CCCC2(CCN(C(=O)CC3(O)CCCOC3)CC2)C1 c1(C(=O)NC(CC(C)NC(C2CCCC(C(N)=O)C2)=O)C)ccc2[nH]ccc2n1 c1(CC)cccc(C(c2nnnn2CC2CCCO2)NC2CCC(=O)NC2)n1 CCCCCCCCc1cn(C(C)C(C23CC(NS(=O)(=O)c4cccs4)(C2)C3)=O)nn1 CC1=NS(=O)(=O)N(C)C=C1C(=O)N(CCCNC(=O)C(C)Cn1cccn1)C N1(C(C(C)C(C)(C)C)=O)CC(C(=O)NOC2CCCC2)CC12CCC2 CC1(C)CN(C(=O)C(=O)NC2CCN(c3ccccc3C(F)(F)F)C2=O)CCN1 c1(Cn2cc(C(C)(C)OC)nn2)ccc(-c2ccc(Br)cc2)cc1 N1(C(C(c2ccccn2)C)=O)CC=CC(C(=O)NCCc2cc[nH]n2)C1 c1(C(N2CCC(NC(=O)Cc3ccon3)C(F)C2)=O)ccc2n[nH]cc2c1F c1(C(=O)NCC2CN(C(=O)CC3CCCC3)CC2O)ncc(Cl)cc1F C12(NC(c3cnco3)=O)CCCC1N(C(=O)CCc1c(F)cccc1Cl)CCC2 CCC(C)CC(=O)NC1CC(c2ccccc2)(NC(=O)CC2CNC(=O)C2)C1 N1(C(c2c(CNC(CN(C3CCC3)CC)=O)ocn2)=O)CCNC(=O)CC1 C(C)(C(=O)N1CC(C(=O)NCCNC(=O)C(C2CC2)SC)C1)SCCCC c1(CC)c(C(=O)NC2CC(F)(CNC(C3CC3(C)C(F)F)=O)C2)cnn1CC C1(O)(CCNC(C2C(CC)C2)=O)CCN(C(C2CCCOC2)=O)CC1 C1(CC(=O)N(C)Cc2cn(CC)nn2)CCCCN1C(c1cn(C)nn1)=O N1(C(C2CCN(C)O2)=O)CCC(CN(C)C(c2cc(C3CC3)nn2C)=O)CC1 C#Cc1cc(C(=O)NC2COCC2NC(=O)CCc2cnc(C)s2)ccc1Cl N1(CC(=O)NC2C(NC(C(=O)NCC)=O)COC2)C(=O)NC(C)(C2CC2)C1=O C1(F)(NC(=O)NC(C)CNC(=O)NC2CC2)COCCN(C(c2ccccc2)=O)C1 CC1(C)OC2CN(S(=O)(=O)c3cccc(CC(=O)O)c3)CC2O1 c1(OC)ccnc(NC(C2CCN2C(c2cccc(F)n2)=O)=O)c1I CCC(CNC(C1CN(C)CCO1)=O)(CC)C(=O)NC(c1cccc(C)n1)C C1(C(=O)OC)CN(CC(c2nc(C3CC3)cs2)=O)CC1C1CCOCC1 C(=O)(C#CC1CCC(=O)CC1)NCCN(C)C(c1ccc(CNS(C)(=O)=O)o1)=O c1(CNC(C(C2CN(C(C3(N(C)C)CCC3)=O)C2)OC)=O)ccc(CO)c(F)c1 c1(C(=O)NC2CC(C)(COC)N(C(=O)C=CCO)C2)cc(C)c(C)nc1C C(=O)(C(C)NC(=O)CN(C1CN(C(=O)CCC2CCCC2)C1)C)NC(C)C S1(=O)(=O)c2ccc3c(c2)SC(=NCCC(CC)(C)N1C)N3.C(C)(C)(CC)OC N1(C(CC)=O)CCCC(N(C(=O)C(O)Cc2ccccc2)CCF)C1 C1(NC(C(COCC)C)=O)CCCCC1NC(=O)Cc1cccc(Cl)c1 C(=O)(C(C)(C)CC#N)N(C)CC1CCCCC1NC(=O)CCCc1ccsc1 c1(C(N(CCNC(C(C(=O)OC)OC)=O)CC2CC2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(N(C(c2cc(CC)on2)=O)C)CCCN(C(=O)C=Cc2nccs2)C1 c1(CC)ccc(C(=O)NC23CC(NC(c4cn(CCSC)nc4C)=O)(C2)C3)cc1 CCC(CC(F)F)C(=O)N1CCCC1(C)CNC(C1CC2CCC(C1)N2C)=O C(CC(=O)NCCCN(C)C(c1cc(Br)cnc1S)=O)(C(C)C)OCC C(=O)(C1CCCn2cnnc21)N1CCCN(C(C(C#C)(C)C)=O)CC1CO c1(NC(c2cc(C)[nH]c2)=O)nc2c(s1)CC(NC(c1nc(C)n(C)n1)=O)CC2 c1(OC)cccc2c(CC(N3CCC3CNC(=O)C(F)(F)F)=O)c(C)[nH]c12 n1(CC)nc(C(=O)N(C(CNC(=O)CCF)C2CC2)C)c(=O)c2ccccc12 C=C(C)CC(C(=O)NCCc1cc(C(=O)NCC(C)C(=O)OC)no1)OC c1(C(N2CC(CCNC(CCCCCC#C)=O)C2)=O)cc2cc(C)ccc2[nH]1 c1(CC)ccc(C(N2CC(NC(=O)CC3(CO)CCCC3)C3(CC3)C2)=O)c(Cl)c1 c1(C(=O)NC2C(CNC(=O)CSc3cccnc3)CC2)ccc(F)cn1 CCC(CCC(=O)NC(C)CCCC1CC1)NC(=O)CC(C)(C)COC c1(C(C)NC(C(=O)NC(c2ccccc2)C(=O)OCC)=O)cccc(Br)c1F N1(C(CN(CC(C)Nc2ccccc2)C)CBr)CCOCC1 CC1CCCC(CCNCC(c2ccc(O)cc2)O)C1 N1(C(C=C(CCC)C)=O)CCC(NC(c2cccc(OC)n2)=O)CC1 c1(C(=O)NC2CCC(CNC(C(N)=O)=O)C2)cccc(CF)c1 N1(Cc2c(C(=O)O)[nH]cn2)CCC(CO)C12CCOCC2 c1(C(=O)NC2CC(C)(NC(=O)CCCF)C2)cccc2c1OCC2 C1(NC(C2C(=C)C2)=O)CCC2CN(c3cc(C(=O)OC)nc(C)n3)CC2C1 Cc1nc(C2CC2)oc1C(=O)NC1CN(C(C2(Cl)CC2CC(C)C)=O)CC1O CN=C1NC2=NC(C3(C)CC3)CC(CF)N=C(N2)N1.c1ccccc1Br n1(CCN(C(C(C)OC2CCCC2)=O)C)cc(C2C3CCCC23)nn1 C(CCCO)(C(C)(C)C)OC(=O)NC(C)CCC(=O)Nc1ccccc1 CC#CCC(C(=O)NOCCCCC1CC1)NC(=O)C(CC)CCCCC C(=O)(C(C)S(N)(=O)=O)NCCC(C)NC(c1ccnn1-c1ccccc1)=O c1(CC)nc(C)ncc1C(=O)NCC(C)(C)CN(C(=O)CC1COCC(C)O1)C C1(C(N2C(CNC(c3nc(-c4cn(C)nc4)sc3)=O)CCC2)=O)CCCC1(C)C C(CCC(O)C(=O)N(CC(N)=O)C)NC(c1c(CC)cns1)=O C=CC(C)(CCOC)C(=O)NCC1(NC(c2ccnnc2)=O)CCCCC1 N#Cc1cc(CNC(C2COCCN(C(C3CC34CC4)=O)C2)=O)cc(Br)c1 Cc1cc(F)ccc1C(=O)NCC(N1CCC(O)C(NC(C(N)=O)C(N)=O)C1)=O N1(C(C(C(C)C)NC(N)=O)=O)CCC(NC(=O)C=Cc2ccsc2)C2(CCC2)C1 C1(CNC(CN(C(C(c2ccn(C)n2)C)=O)C)=O)CCN(C(=O)CO)C1 c1(OC)cc(NC(C2OCCC2CNC(C2CC(=O)NC(=O)C2)=O)=O)ccc1F N1(C(c2cc(C#N)no2)=O)C2CCC1CC(NC(=O)CN1CCCC1CO)C2 c1(C(C)C(N2CC(O)(CNC(C3CC3c3ccco3)=O)C2)=O)cc(F)cc(F)c1 C1(CC(N2CCC(C)(CNC(c3ccsc3C#N)=O)C2)=O)(OCC)CCOCC1 CC(C)C(N=[N+]=[N-])C(=O)N(CC(N1CCC(N2CCC2)C1C)=O)C N1(C(C2C(OCC)C2)=O)CCOCC(CNC(C2CCSC2)=O)C1 c1(CC)n[nH]c(CC)c1CC(=O)NC(C)(C)CNC(=O)CC1CCC12CCC2 c1(C(=O)NC2CC(CNC(CCSCCC)=O)C23CCC3)ccn2ccnc2c1 CCC(F)(F)C(=O)N(CC(O)CNC(c1cscc1C(F)F)=O)C C1(NC(c2cc(N)cc(O)c2)=O)CC(NC(c2cnsc2)=O)C12CCOCC2 c1(NC(C(C)C)=O)ccc(F)cc1NC1(c2nnnn2CC2CC2)CCC(C)C1 N1(C(C2(F)C(C)C2)=O)CCC(N(C(=O)CSc2ccccn2)CCO)C1 C1(NC(C(C)NC(c2ccco2)=O)=O)CC(C)(NC(C23COCC2C3)=O)C1 N1(C(CCNC(C2CCN2C2CCCC2)=O)=O)CCC(CCOCC)C1.C1CO1 CC(N=c1[nH]nc(O)s1)C1CCCN(C(C2CC(O)CN2C(N)=O)=O)C1 C(C)(CCCCN=c1[nH]cnc2cc(C3CC3)nn12)OC.c12sccc1C(=O)NC2 N1(C(C(n2cc(C)nc2)(C)C)=O)CC(C)N(C(=O)Cn2cccc2)CC1C CC1(C)COCCC1NC(=O)CNC(=O)CC1CC=CCC1 c1(C(=O)NCC(C)(C2CCC2)NC(C(F)=CCC)=O)nsnc1O C(=O)(C(O)COC(=N)O)N1CC(C(C(=O)NCC(C)(O)c2nn[nH]n2)O)C1 C(=O)(C(C)CCCC)N(CC(=O)NCCNC(=O)NC)CC#C C1(C(=O)NCC(CC)n2cccn2)CC2CN(C(C3COCCN3C)=O)CC2C1 Cc1nonc1CC(=O)NC(CN(C(=O)C(O)CN(C)C)C)Cc1ccccc1 C12(C(=O)NC3C(OC)CC3O)CC(CN(C(c3cn(C4CC4)nn3)=O)C1)C2 n1(CC(=O)N(CCOC)C)ccc(=NCc2ccc(OCC(C)C)cn2)nc1O C(=O)(C(C)(C)C(C)(F)F)N1CCC(NC(C(C)OC2CCCCCC2)=O)C(F)C1 c1(C(=O)NC2Cc3n(cc(C)n3)CC2)ccc2c(c1)CNC2=O c1(C(N(CC(C)N(C(C(CC)F)=O)C)C)=O)cncc(N2CCOCC2)c1 CC1CC(NC(c2ccn(-c3ccc(F)cc3)n2)=O)CCN1C(C1(C#N)CC1)=O c1(CNC(C(c2cccnc2)NC(CCCNC(=O)OC)=O)=O)cccc(C)n1 N1(C(C2N(C(C(CC)n3ccnc3)=O)CCC2)=O)CCC(CC2CC2)CC1 c12ccc(Cl)cc1-c1csc(n1)C(=O)N2.N12CCCC1(C)C2.Cc1ncc(C(C)C=O)[nH]1 N1(C(=O)NC(C2C(c3ccc(CC)cc3)C2)=O)Cc2ccccc2CCC1CC Cc1cccc(C)c1NC(=O)C(N1CCCC(C(C)(F)F)C1)c1cncs1 c1(C(N2CC3C(NC(c4nncs4)=O)C(C3)C2)=O)ccc2cc(Cl)ccc2c1 C1(NC(CS(CC)=O)=O)CCCN(Cc2ccn(CC(C)C)n2)CC1 N1(C(C2CC3C=CC2C3)=O)CCC2(CC1)CCN(C(C1CC3(CCO1)CC3)=O)C2 C1(C2CN(C(c3ccc(Br)c(CO)c3)=O)C2)(NC(CC2(C)CCCO2)=O)CC1 CCCC(CCC)CC(=O)N1CC(O)CC1CNC(=O)CC1(CO)CCOCC1 c1(NC(C=CC2N(C(=O)OC(C)(C)C)CCC2)=O)cc(Br)ccc1O C1(C(C)C)CN(C(c2cn(CCCF)nn2)=O)CCN1C(=O)CN(C)C1CC1 C1(C(N(C(CC)C2CC2)C)=O)C=CCCN1C(=O)C(C)CSC C1(NCc2scc(C)c2)CC(NC(c2ncoc2-c2cccs2)=O)C12CCC2 c1(CN(C)CCN2CCOC(C)(c3ccccc3)C2)nc2cc([N+](=O)[O-])ccc2o1 Cc1ccc(NC(=O)COCCOCF)c(OC)c1.C1(NC)CCOC1 C=C1CCN(C(=O)CC2CCOCC2)C(C(=O)NC2COC3(CCC3)C2)C1 Cc1c(Cl)ccnc1C(=O)NC1CC12CC(NC(C1CC(F)C1)=O)C2 C1(C(=O)NCc2c(C)nn[nH]2)CN(C(C2(O)CCCC2)=O)CCN1C C(Cc1cc[nH]n1)(C(=O)NC(C)COC)NC(C=CCN(CC)CC)=O C1(NC(C2(CC)CC2)=O)CCCSC1.C(CCC(C)C)OCC(=O)N1N(C2CC2)C1 c1(OCC)ccc(C)cc1CNC1COCCN1C(=O)Cc1cccnc1Br c1(CC(=O)Nc2n(C)nc(C(=O)OCC)c2Cl)c(F)cccc1C#N C1(C(N2CC(C(N)=O)(CNC(c3sccc3F)=O)C2)=O)CC(C2CC2)=NO1 N1(Cc2cc(C)n(C)n2)CCC(O)C(C(N2CCC(C(C)(C)C(=O)O)CC2)=O)C1 n1(CC)cc(Cl)cc1C(=O)NCCC(C)NC(=O)CC1CC2(CC2)CO1 c1(C(=O)NC(C2CC=CCC2)C(=O)NC(CCCCC)C)c[nH]c(C#N)c1C CCC(C(=O)NCC(C)CN(C)C(c1ccc(C(F)(F)F)o1)=O)C(C)O c1(C(=O)NCC2N(C(CCOCC)=O)CCC(C)C2)cc2c(nc1O)CCSC2 c1(CCC)cc(C(=O)NC2(C)CCN(C(c3coc(N(C)C)n3)=O)C2)n(C)n1 CCCCC(O)CC(=O)NCC1(CCNC(=O)C(CC)c2cccnc2)CC1 c1(OC)cccc([N+](=O)[O-])c1CN1CCNCC1C(=O)Nc1ccnc(C#N)c1 C=CC1(CNC(N2C(C(=O)NCC3CCCCC3)CCC2)=O)CCC1 c1(C(=O)NCC(CC)NC(c2cc(C)[nH]n2)=O)cccc(C(N)=O)c1C Cn1ncc2c1CN(C(=O)CC1CC(F)CN1C(C1CC=CCC1)=O)CC2 C1(NC(c2nc(C)sc2)=O)C(C)CCN(C(C2CCCCN2C)=O)C1C N1(C(c2cnn(C)c2Cl)=O)CC(NC(c2ccc(C3CC3)o2)=O)CC12CCC2 c1(C(=O)NCC(CCNC(=O)Cc2cnc[nH]2)O)occ2c1CCOC2 C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC1N(C(CC(C)(C)C)=O)CC(F)C1 C1(CC(N2CCC(CC=C)(NC(=O)C(C)=CC(C)(C)C)C2)=O)CCC(C)(C)CC1 N1(C(C2CC2CF)=O)CCOC(CNC(=O)C(F)(F)CC(C)(C)C)C1 C1(NC(c2c(C)sc(O)n2)=O)CCN(c2snc(Cl)c2C#N)CC1C Cc1ccc(C(N2CCC(NC(c3ncc(F)cc3C)=O)C(C)C2)=O)c(F)c1 C1(C(=O)NCC2(OC)CCC2)(NC(=O)CCC2CC(F)(F)C2)CCCC1 C12(C(N3CCC(N(CCC)C(C4(C)CCCC4C)=O)CC3)=O)CCCN1CCC2 C1(C2(O)CN(C(c3cc(Cl)cn3CC)=O)C2)(CNC(C(C)SCC)=O)CC1 C1(NC(C(C)(C)O)=O)CN(C(c2cc(C3CC3)nc(Cl)c2)=O)CCC1C(F)(F)F C1(C)(c2cn(CCC(=O)OC)nn2)CCCC(CN)C1 c1(C(N2C(C)CC(NC(C3(CC)CC3)=O)C2)=O)ccc(C)c(C(C)(C)C)c1 c1(OC)ccc([N+](=O)[O-])c(N2CCC(NC(c3nc(C)sc3C)=O)C(O)C2)n1 c1(C(=O)OCC)c(C(C)(C)C)csc1C(=O)NC1(C)CC(C)=NO1 N1(C(C(C)OCC)=O)CCOC(CC(=O)NCc2cn[nH]c2)C1 C(=O)(CC(COC)COC)NC(C(=O)NCCn1c(CC)ncc1)COC c1(CC2CC(c3cn(-c4cccc(C(=O)O)c4)nn3)C2)nc(Cl)ccc1Br N1(C(=O)Nc2ccc(OC)nc2)CCc2c(ccnc2OC)C1 Cc1noc2ncc(C(=O)NCC(CO)NC(=O)CC3(O)CCCOC3)cc12 C(=O)(C(F)CCC(C)(C)C)N(C(=O)C(N1CCCC1)C1CC1)C(C)Nc1cccnc1 N1(C(CC(C)(C)SC)=O)CCC(C2CCOCC2)(CNC(=O)C(C)C(C)O)C1 C1(NC(C2(COC)CCCCC2)=O)CC(O)CN(C(=O)CCN2CCC(F)C2)C1 C(=O)(C(=O)C(C)(C)C)N1CCC(N(C(=O)CC2CCNC(=O)C2)C)C1 CC(CC(N)=O)C(=O)NCCOCCN(C(=O)Cc1ccco1)C Cc1ccc(C(=O)N(CC(=O)NC(c2cccnc2F)C)C(C)C)cc1[N+](=O)[O-] c1(OC)ccc(C(N2CCCC(C(=O)NCCN3CCCC(C)C3)C2)=O)cc1I C1(=CC(=O)NCCOCCNC(C2CCC(C)CO2)=O)CCCCC1(C)C C1(C)(C(=O)NC)CCN(C(c2sc(Br)nc2Cl)C(=O)NCCCC2CC2)C1 c1(C(=O)NCCNC(C(C)(C)C2CCOC2)=O)ccc(C2=CCCC2)cc1 N1(C(C(CC)SC)=O)CC2(CC(NC(C3CC3C(F)F)=O)CO2)C1 C1(CNCCC(=O)NC(c2c(NC(C)=O)cccc2)=O)CN(C)CCC1O Cc1cncc(C(=O)N(CCCNC(=O)CNC(=O)C=Cc2cccnc2)C)n1 C1(CN(C(=O)CN2C(=O)CCC2=O)C)CCCC(NC(=O)CC2(CO)CC2)C1 c1(C(=O)NCC(CNC(c2nc(CC(C)C)sc2)=O)CO)ccnc(C2CC2)c1 C1(CNC(=O)CNC(=O)CCF)(NC(=O)C2CC2)CCN(CC(c2ccco2)=O)CC1 c1(C(=O)Nc2c(C)nc(Cl)nc2)cc2c(-c3ccc4oncc4c3)cncc2s1 N1(C(C2OCC(C)C2)=O)CCCC2(NC(=O)C=Cc3cccc(F)c3)CCCC12 N#CC1CC(C(N2CCC2C2CCOCC2)=O)C1.C1(N2C(=O)C2)CCCCC1 C1(C(N2CC(CC(C)NC(=O)CSCC#N)C2)=O)CCOCC1C Cc1ccc(C(N2CCC(C)(NC(c3sc(=N)[nH]c3C)=O)CC2)=O)nc1O Cc1ccc(C=CC(=O)N(C)CC2CCCN2C(c2cc(C(F)F)cs2)=O)s1 c12cc(c(F)cc1[N+](=O)[O-])NC1CCN2C1.C1(C(C)C)CCCC1OC.CO CC(CN(C)C)CCC(=O)NCCCNC(C1(C(F)(F)F)CC(F)(F)C1)=O Cc1oc([N+](=O)[O-])cc1C(N1CCCC(O)(CNC(=O)CC2CCCCO2)C1)=O CC1(C)CN(C(=O)C(C)(F)c2ccon2)CC1NC(C1CCCS1(=O)=O)=O Cc1cc(C(=O)NCC2CCC(NC(C3CC=CC3)=O)C2)c2nc(C)n(C)c2n1 N1(C(C(CCSC)O)=O)CC2C3CCC(C2C1)N(C(c1cccc(F)c1C)=O)C3 S(=O)(=O)(c1ccc2[nH]c(=NC(C)C(C)C)sc2c1)Nc1c(CC)n(CC)nc1 C1(C2CCCN(C(C3CC4C(C3)C4(C)C)=O)C2)(NC(C(CCSC)OC)=O)CC1 C(=O)(C(C)CC(C)CC)N(C(C(=O)N1C(C(N)=O)CC(OC)C1)CC(C)C)C N1(CC#N)CCCC(CNc2c(-c3ccccc3)ncn2C)C1 N12CC(CC13CCC3)SCC(O)C2=O.C(=O)(CNC)N(C1CCC1)CC.OC c1(C(=O)NC2CCC(N(C(=O)COCc3nc[nH]n3)C)C2)cnc(S)nc1 c1(CC(=O)NC2CC(CNC(CCN(C)CC)=O)C2(C)C)c(C)nn(C)c1Cl N1(C(c2c(C)con2)=O)CCCCC1CNC(=O)C(c1cccc(Cl)c1)N(C)C Cc1oncc1C(=O)NCCC(N1CC(F)(CNC(c2csc(Cl)n2)=O)C1)=O Cc1ccc2snc(C(=O)NCC(O)CNC(=O)CC3CC3(C)C)c2c1 c1(C2(C(N(CCCNC(C3(C)CCC3)=O)C3CC3)=O)CC2)cc(F)ccc1F c1(C(N2CC(O)(CNC(c3ncccc3F)=O)C2)=O)cc(F)ccc1F C1(OC)CCC2(C(=O)NC3CC(NC(=O)Cn4c(C)csc4=O)CC3O)CC12 Clc1cc2c(N3CCN(CCc4cccc(Br)c4)CC3)ccnc2s1 C(=O)(CCC(O)C(C)(C)C)N1CC(C(=O)NCc2c(C)ccnc2)C(C)(C)CC1 N1(C(CCc2nc(C)sc2)=O)CCC2(NC(=O)CSCCC#N)CC2C1 C1(CCC(=O)NC2CC(n3cncn3)C2)(NC(CNC)=O)CCCC1.C1(C)CC1 c1(NC(C2N(C(c3cc(SC)ncc3)=O)CC(O)C2)=O)ccc2c(c1)CC(=O)N2 c1(CC)cc(C(=O)NCC(c2ccccc2)N(C)C(C2CCCCS2)=O)ccn1 c1(CC(N2CCCN(C(C(C)OC)=O)C(C)C2)=O)ccc([N+](=O)[O-])cc1F C1(NC(C2NC(=O)OCC2)=O)CCN(Cc2ccccc2)C2(CCC2)C1 N1(C(CC2C(NC(C3(C(C)C)CC3)=O)CCC2)=O)CC2CCCCC2C1C c1(C(C(=O)NC(C)C)N(CC(C(C)C)OC)C)ccc(-c2ccco2)cc1 N1(C(C2C(=C)C2C(=O)OC)=O)CCCCC1CC(=O)N(C)CC1CCOC1 CC(O)(C(=O)NC1CCC(CC(=O)NCC(O)C(N)=O)C1)C(F)(F)F c1(NC(c2ncc[nH]2)CC)cc(N2CCN(CCCC3CCCS3)CC2)ncn1 C12(NC(C3C(C=C)OCC3)=O)CCC(C1)N(C(=O)Cc1n[nH]c(=N)s1)C2 c1(CC)nc(C)[nH]c1C(=O)NC(C1(O)CCN(C(=O)C=C(C)C)C1)C C1(NC(c2cnc(OCC)nc2)=O)CCN(C(C2CCC(=O)NC2)=O)C12CC2 C1(NC(C2CCCN2C2CCCC2)=O)C2CC1CN(C(c1ccccc1F)=O)C2 CC1CCCCN(C(C2CC(O)CN2C(=O)CN2CCCCC2C)=O)C1 Cc1nc(C(=O)NCC2C=CC(NC(=O)C(C)CC(C)(F)F)C2)c2ccccn12 c1(NC(C(C)C)C(C)NC(c2cc3n(n2)CCO3)=O)ncnc2scc(Br)c12 C(CC(C(C)C)NC(c1ccnn1C)=O)N(C(C(C)NC(C)=O)=O)C N1(C(C(N2CC(C)C2)C)=O)C2CCC1CC(C(=O)NCc1ccncc1Cl)C2 C1(NC(=O)COCC2CC2)COCC1NC(=O)COCC1CCCC1 C1(C(N2CCN(CCNC(C(CN(C)C)O)=O)C(=O)C2)=O)CC2OC(=O)OC2C1 c1(C(N2CC3C(CNC(C=C(c4cn(C)nc4)F)=O)C3C2)=O)ccc(N)cc1O C1(CC)CCCN(CC(=O)NCC(C)(O)CNC(=O)CCCN2CCCC2)C1 [N-]=[N+]=NCCCCC(=O)N1CC(=C(F)CNC(=O)CCCCN2CCCC2)C1 CCCC(F)(F)C(=O)NCC1OCCC1C(=O)Nc1csc(C)c1 C(=O)(C(CC)CC(F)(F)F)N(CCC)CCNC(c1c(C)coc1C)=O Cc1cc(C#N)ccc1C(N1CC2CCC(NC(C3CC3[N+](=O)[O-])=O)(C2)C1)=O CC1CN(C(=O)CC2CCCSC2)CC(C(=O)NCCC2NC(=O)NC2=O)O1 c1(C(=O)NC2CC(CNC(Cc3n(C)ccc3)=O)C2)cc(F)c(CO)c(F)c1 C(CS(=O)(=O)c1cccc(C(F)(F)F)c1)N(C(C1CCN1C1CCCC1)=O)CCO c1(C(N2CCC(N(C(CSCC)=O)CC)CC2)=O)ccn2cnnc2c1 N1(C(c2c(SC)ccc(N)c2)=O)CC2(CCN(C(=O)C(c3nc(C)cs3)C)C2)C1 c1(-c2n(C3CCCC(C)C3)nc(-c3ccc(F)cc3)n2)ccc2c(n1)CCCC2 N1(CCS(CC)(=O)=O)CCC2(CC1)CCN(C(=O)CN1CC(=O)NC1=O)CC2 C(c1ccc(C)o1)=CC(N1CCC(C(N2CCC(CC)C2)=O)C1)=O O(NC(=O)C(C1(O)CCC1)NC(=O)C(C)N(CC)CC)C(C=C)C c1(NC(c2c(-c3cc(OCC)c(CC)cc3)ncs2)=O)cccc(F)c1[N+](=O)[O-] CCCC(O)CC(=O)N1CC(NC(=O)COC2CC(F)(F)C2)C2(CCC2)C1 C=C=CCCC(=O)NC(C)(CNC(=O)CSCCN(c1ccc(F)cc1)C)CO N1(C(C2(C)CCSCC2)=O)CCC(NC(c2n[nH]c(C3CC3)c2Cl)=O)CC(O)C1 c1(N(CC(C)(C)CO)C)nc(=N)[nH]c(=NCC2CC(C)(C)CCC2O)[nH]1.C(C)(C)C Cc1n[nH]c(C)c1SCC(=O)NCC1C=CCN1C(c1cnc(C(C)C)nc1)=O N1(C(C(C)NC(CC)=O)=O)CC2(CCCN(C(C3CCCC(O)C3)=O)C2)C1 N1(C(C2(NC(C)=O)CC2)=O)CC(NC(=O)Cc2csc(C3CC3)n2)CC(O)C1 N1(C(c2cc(C)no2)=O)CC2(CC(CC(=O)N(C)Cc3scnc3C)C2)C1 c1(C(N(CCC(N2CCC(CSC3(C4CC4)CC3)C2)=O)CC)=O)cccc(CSC)c1 N1(C(C2(C)C(C)OCC2)=O)CCC2(CC1)CC2C(=O)NCc1nn[nH]n1 Cc1cc(F)ccc1C(O)C(=O)NCC(C)N(C)C(c1ccnn(C)c1=O)=O N1(C(C(CC)CC)=O)CCC(C)(C)C(C(=O)N(CCCC(O)CO)C)C1 CC1CN(CCO)CC(C)N1C(=O)CCCn1cc(C2(C)CSC2)nn1 Cc1ccc2[nH]nc(C(=O)NCC3CCN3C(=O)C(C3CC(F)(F)C3)O)c2c1 C1(c2nc(C(C)C3CC3)nn2-c2cnn(C(C)C)c2)Cc2ccccc2N1C C1(NC(c2c(CC)cc(N)cc2)=O)CCCCCN(C(=O)C(F)C2CCC2)C1 c1(C(C(=O)N(C)CC2CCCCC2N)(F)F)cccc(Cl)c1Cl C(=O)(C1=Cc2cc(F)ccc2OC1)N1CC2C(CCNC(C(F)=CC)=O)(CC2)C1 N1(C(CC(C)F)=O)CCC2CCCC(C1)N2C(c1cccc(Br)c1F)=O C(CS(=O)(=O)CC(=O)N1CC2CCC2(CC(=O)NC(c2cnsc2)C)C1)OC C1(C(=O)NCC(C)C(=O)NC2COC(=O)C2)OC2CCC1C2 N1(C(C)C)CCCCC1C(=O)NC1(CCNC(=O)CC2CCC(=O)N2)CC1 C1(NC(C(c2n(C)ccc2)=O)=O)CN(C(=O)CC=C(Cl)Cl)CC12CCC2 CC1=NOC(=O)C1CCC(=O)NCC(C)N(C)C(c1ncccc1C(C)(C)C)=O N1(C(CCOC(C)C)=O)CCC2CN(C(c3cccc(=O)o3)=O)CC2C1 C1(NC(c2cc(C)nc(O)c2)=O)CN(C(c2c(C)ccn2C)=O)CC(C)(C)C1 Cc1ccn(CC(=O)NC(C)(CNC(=O)Cc2nnc(O)s2)CC(C)C)c(=O)c1 Cc1c(C(N2CCN(C)CC2CNC(=O)CC2CC2C2CC2)=O)cccc1Br C(=O)(C(C)CC(C)C)N1C(C)(C(=O)NCC(CC)(C)CC)CCC1 N1(C(CC2CCC(C)(C)O2)=O)CC2(CCCC2)C1C(N1CC2CC2C1)=O C(=O)(C1COc2ccccc21)NC1(CNC(C(C)(Cl)Cl)=O)CC2CCC1CC2 C1(NC(CCn2c(C)ncc2)=O)CN(C(C2CC(C#N)C2)=O)CC12CC2 N1(C(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC(O)C1 C1(C(N2CC(F)(F)C2C2CC2)=O)CC2CCC1N2C(C1COCC1C(F)F)=O Cc1cccc(CNC(=O)C(C2CC2(C)Br)N(CC(=O)NCC2CC2)C)c1 CC1CN(C)CCCN1C(c1cccc(-n2cc(C(N3CCCC3)C)nn2)c1)=O C1(C(N2C(C(C)NC(Cc3c(C)cccc3)=O)CCC2)=O)CCC2(CC1)CC2 C(CC(=O)N1CCOC2CC12)(C(C)C)NC(c1c(C)snc1)=O CC(C)C(F)(CNC(C1CC2CC1CC2=O)=O)C(=O)NC(C)C(O)C(F)F C#CCC(CC)NC(c1sccc1CNC(=O)CCOCC1CC1)=O C1(O)(CN2CC3CCCN(C(C4N(CC)CC4)=O)C3C2)CCc2ccccc2C1 Cc1ccc(F)c(C(C)NC2CCC(N)C2)c1F C1(CC(=O)NC(C2N(C(Cc3c(C)occ3)=O)CCC2)(C)C)CCS(=O)(=O)C1 Cc1cc(C(=O)O)cc(C)c1NC(c1ccc(CN(C)C)c(F)c1)=O C(CS(=O)(=O)CC(=O)N(CCCC(=O)NC(CCO)C1CCCC1)C)OC c1(C(=O)NC(C2(C(N3C(C#C)CC3)=O)CC2)C)sc(F)cc1C C(CCCCCNC(C1CCOC(=O)N1)=O)NC(CNS(N)(=O)=O)=O N1(C(Cc2c(C)cccn2)=O)Cc2occ(C(=O)NCCCC(F)F)c2C1 CS(=O)(=O)c1cnc(N2CCC(C3CCCCN3C(C3CSC3)=O)C2)c(Cl)c1 N#Cc1cnnc(N2CCOCC2)c1.C12(F)CC(C1)C(=O)NC2 C=CCC(C(=O)N1CC(NC(=O)CNC(=O)NC2CC2)CCC(O)C1)C(C)C C12(NC(C=CCOC)=O)CCC(C1)N(C(C1(C3CC3)CC=CC1)=O)C2 c1(SC)nc(O)c(C(N2CC(NC(C3CCC(O)C3)=O)C2)=O)cc1C#N CCCC(C)C(C)NC(N1CCN(C(=O)OC)CC1)=O N1(C(c2scc(OC)c2)=O)CC(OC)CC1C(=O)NCCSCCO C1(OC)(CNC(c2ccnc(Cl)c2F)=O)CCN(C(=O)C(=O)NC2CC2)CC1 c1(NC2CCC(CCC)CC2)ccc(S(=O)(=O)N2CCCCC2C)c(OCC)c1 C(N=c1ccc2cc(S(=O)(=O)c3ccccc3O)ccc2[nH]1)c1c(CC)con1 C#Cc1cc(C(=O)NCC(C)(CO)NC(=O)C(CC)n2ccnc2)cc(F)c1 C1(CNC(CN(C(C)=O)C)=O)CN(C(c2n[nH]c(C3CC3)c2C)=O)CCC1(F)F C1(NC(C(CCC)(C)C)=O)CC2CN(c3nc(C(F)(F)F)cc(C)n3)CC2C1 CN1CCCC2(CCN(C(=O)Nc3cnc4ccnn4c3)C2)C1=O N1(C(c2ccccc2Br)C)C(=O)CCN(CCCc2cccnc2)C1=O N=c1[nH]nc2ccc(N3CCN(c4cc(-c5ccco5)[nH]n4)CC3)nn12 C1(C(=O)NC2C(NC(c3cn(C)nn3)=O)CCOC2)CN2CC3CC2(CO1)C3 C(=O)(N=c1ccn(C(F)F)[nH]1)C1(NC(C(C2CC2)OCC)=O)CCC1 Nc1ccc(-c2cn(CC(=O)Nc3ccccc3C(F)(F)F)nn2)cc1 N1(C(C2(CC)CN(C(=O)Cc3ccc(C)cn3)C2)=O)CCC2(CC1)CC2 C1(S(C)=O)(C(=O)OCC)CCN(C(c2cc(C(F)F)nc3ccnn23)=O)CC1 C12(C(N3CCC(NC(C(N4CCOC4=O)C)=O)C3)=O)CCC(CF)(C1)OC2 N1(C(CC(C)(C)OC)=O)CCC(C(=O)NC2(C)CCC(C)(C)C2)C(C)C1 c1(C(=O)OC)cc(C(=O)NCC=CCNC(C2(C(C)C)CCC2)=O)ccc1C C#CCC(CC(=O)NC1CN(C(=O)COC)CC1NC(=O)OC)c1ccccc1 C(=O)(CC(O)C(C)(C)C)NCC(CNC(CCCN1CCN(C(C)C)CC1)=O)C c1(C(=O)NC2(C(N3C(CNC(C)=O)C=CC3)=O)CC2(C)C)ncn(C)c1C C(=O)(CC(C)CC(C)C)NCC1CCN(C(CCCCC=C(C)C)=O)C(C)C1 C(=O)(CCC(=O)CNC(C12CCCC1CCC2)=O)OC C1(C(=O)NCC(C2(O)CN(C(=O)CNC=O)C2)(C)C)CC12CCCC2 C1(C(=O)O)CN(C(c2cc3cnccc3o2)=O)C2(CCCCC2)C1 c1(NC(N2C(C(=O)NC(C(=O)NCC)C)CC2)=O)ccc(OC)c(C)c1C CCC(C)(C#N)C(=O)NC1CC(O)(CNC(c2cnccn2)=O)C1 C1(C)(C(=O)NC(c2cn(Cc3n(C)cnc3)nn2)C)CCC2(CC1)CC2 C1(CCNC(=O)C(c2ccc(Cl)cc2)CC2CC2)CCCN(C(=O)CO)C1 C1(CC)C(NC(=O)Cn2cccnc2=O)CCCN1C(=O)CC1CCCC(=O)N1 c1(C(N(C)CC2CCCN(C(CC(C)F)=O)C2)=O)cc(N)c(F)cn1 C1(C(N(CC)Cc2cnc[nH]2)=O)C=CC(NC(=O)CNS(N)(=O)=O)C1 N1(C(C2CCC(C)(F)CC2)=O)CC2CCCN(C(C3CN4CCN3CC4)=O)C2C1 n1(CCSCC(C)(C)C#N)c(C(C)(C)C)nnc1Br N1(C(c2c(OC)noc2C)=O)CC2ON=C(CNC(C3(C)CCCCC3)=O)C2C1 C1(NC(c2cccnc2CNC(=O)CCCF)=O)CC(=O)N(O)C1 N1(C(c2ccc(C)nn2)=O)CCC(CO)C(NC(c2coc3c2CSC3)=O)C1 c1(CC(=O)OC)cc(OC)c(OC)c(Oc2ccc(C3(C(N)=O)CCOC3)cc2)c1 N1(C(C(N2CCC(N(C)C)CC2)C)=O)CC(C)CCC1CNC(=O)CCCC#N C(=O)(C1CCCc2cncn21)N1CC2C(Nc3cc(C#N)ncn3)(CCC2)C1 CC1CCC(=CC(=O)NC2CC2CNC(=O)CSCC(N2CCCCC2)=O)C1 CC(CCC(=O)NCCN(C)C(C1CCS(=O)(=O)N1C)=O)S(C)(=O)=O C1(C(=O)NCC(C2CCCS2)C)(CNC(C2CCC(N(C)C)C2)=O)CCOC1 c1(OC)ncc(C=CC(=O)NC2CC3(C2)CN(C(=O)CC2CC2(Cl)Cl)C3)cn1 c1(C(=O)NC2C(NC(Cc3c(C)n[nH]c3)=O)C2)ccc(C(C)C)cc1F c1(CN2C(C(=O)NCC3CCC(=O)NC3)CC3CC32)cccc(Cl)c1O C(C(=O)NCCCN(C(c1cnc[nH]1)=O)C1CC1)(C(C)C)SC c1(C(C(=O)N(C(=O)CCC)CCN(CCCC)C)(F)F)cccc(Br)c1 N1(C(C23CCC(C)(OC2)C3)=O)CCC(C2CC2NC(c2cnc(Cl)s2)=O)CC1 C1(C(=O)NCC(CN(C)CCS(C)(=O)=O)O)CCCN1C(N1CCCCC1)=O C1(CC)CN(C(=O)C2=CCCOC2)CCC1NC(=O)CC1(C)CCOCC1 C12(CNC(C3(CC)CCC3)=O)CC1CN(C(=O)C=C(C)C1CC1)C2 C1(CNC(C2(C#C)CCC2)=O)COC(C)(C)CN1C(c1nc(CC)sc1C)=O c1(C(N2CC(CNC(c3cc(C)cc(O)c3)=O)OCC2)=O)cnc2ccoc2c1 c1(C(N2C(C(=O)Nc3c(C(N)=O)cccn3)CCC2)=O)cccc2c1NCCC2 N1(C(C)(C)C)CC(C(=O)NC2CCC(NC(C3CC3CF)=O)CC2)CC1=O N1(C(c2sc(C)c(C)c2C)=O)CCCN(C(C2CC(F)C2)=O)C(C)C1 C(CC(C)C)(C(=O)N1CCCCC1C(=O)NCC1CCCC1C(N)=O)NC(C)=O C1(C(=O)NCC2(O)CN(C(CCC(C)CN(C)C)=O)C2)CCc2nc(O)[nH]c2C1 C1(NC(C2CCCC(C)C2)=O)CCCCN(C(c2ccsc2Cl)=O)C1 N1(C(c2cc(C)no2)=O)CCN(C(c2cnn(C)n2)=O)C(c2cccc(Cl)c2)C1 N1(C(Cc2cn(CC)nc2C)=O)CCOc2c(C)cccc2C1 N1(c2c(C)cc(Br)cc2)CCC(NC(=O)CCCCN(C)C)CC(C)(C)C1 C1(C(=O)NCC(C(=O)NCCCC(CC)O)O)CCCCC1(C)C c1(OC)ccc(N)c(-c2cn(CC(=O)NC3CC(SC4CCOCC4)C3)nn2)c1 c1(NC(COCC)=O)ccc(O)c(F)c1.C12CN(CCO1)C(=O)CCC2 c1(C(=O)NC2CC(NC(C3C(C)(C)COCC3)=O)C2)cccc2c1CNC2=O C(CCCC(=O)N1CCC(NC(c2cc(C3CCC3)nn2C)=O)C1C)NC(C)=O C1(NC(c2c(C)n(C)nn2)=O)CC(NC(=O)C=C2CCOCC2)C12CCOCC2 C12(C(=O)NCC(CCC)NC(=O)C(c3ccc(OC)cc3)C)CC3CC1C2C3 c1(CCC(=O)N(CC(C)NC(=O)C=CSc2ccccc2)CC)ccccc1Cl Cn1ncc(S(N)(=O)=O)c1C(=O)NCC(O)CNC(c1ccnn1C1CC1)=O Cc1cc(C)cc(C=CC(N2CCOCC2CCC#N)=O)c1 Cc1c(CC(=O)NCC2CN(C(=O)C(C)CO)C2)c(O)nc2ccccc12 c1(C(CNC(=O)COCc2cnoc2)NC(C2C(CC)C2)=O)ccccc1 C1(c2nnnn2C2CC2)(NC2(SC(F)(F)F)COC2)CCC2CC12 N1(C(CCC)=O)CC(C)(C)C(NC(c2ccc(CC)o2)=O)C(C)(C)C1 C1(O)(CNC(C(c2ccccc2F)OC)=O)CCCCC1 C1(CCNC(C2CC=CCC2)=O)CCCCN1C(=O)Cc1ccsc1Cl C1(C(=O)NC2CCCN(C(C(CCC)=CCC)=O)C2)CN2CCC1CC2 C1(NC(Cc2ncc(CC)[nH]2)=O)CCCCN(C(=O)Cc2nccn2C)C1 C(C#Cc1cnn(C)c1)NC(CC(C(C)C)NC(C(COC)(C)C)=O)=O C1(CNC(c2c(C)scn2)=O)CCN(Cc2cc3sccc3s2)CC1(F)F c1(OC)cc(C(=O)NCC(CC(=O)O)c2ccncc2)ccc1OC(F)F C=CC(C)CC(=O)N(C)CCN(C)C(c1ccnc(OC)n1)=O C(=O)(CCCCC(=O)N1CC(O)(CNC(C2CC(F)(CO)C2)=O)C1)NC N1(C(c2c(Cl)cn(CC)n2)=O)CC(NC(c2sc(F)cc2C)=O)CC2(CC2)C1 c1(CC(=O)NCC(CN(C(C(CC)OCC)=O)C)C)cccc2cccnc12 C=CCC(C)(C)CC(=O)N(C1CCC(NC(=O)CCCCN(C)C(C)C)C1)C C1(C(=O)NCCCCNC(c2c[nH]nc2F)=O)CCn2c(Br)cnc2C1 N1(C(c2ccc(Cl)c(C)c2O)=O)CCOC2(CCN(C(=O)CC(F)(F)F)CC2)C1 c1(CC(=O)NC(C)CCNC(C2CCCC2C)=O)ccc2c(c1)ncn2C Cc1cnc2c(C(N3CC(N(C)C(c4cnc(Cl)[nH]4)=O)C4(CC4)C3)=O)cccn12 C1(CC(C)NC(C2CC2C#N)=O)CCN(C(C2CC(F)(CO)C2)=O)CC1 C=Cc1ccc(C(=O)NC(CNC(=O)CC2CC(CC)C2)C(C)C)cc1 CC1CCN(C(c2cnn(CC(F)F)n2)=O)CC1CNC(=O)CSC1CC1 N1(C(C2CCN(CC)C2)=O)CCC2(CC1)CC2(C)C(=O)N(c1ccccn1)CC C1(C)(C(N2CC(CNC(CC3(C)CC3)=O)C(O)C2)=O)CCCS1(=O)=O c1(SCC(=O)NC(C(CO)NC(C2N(C(C)=O)CSC2)=O)C)cccc(Cl)c1 c1(CCN(CCN(C(C(C)OCC(=O)OC)=O)C)C)sc(CC(C)C)nc1C C12(C(N(C3CN(C(C4(O)CCCCC4)=O)C3)C)=O)C3C4C1C1C2C3C41C#N C(=O)(CCS(C)=O)NCC(CN(C)C(c1[nH]cnc1C#N)=O)(C)C c1(N2CC(CCCCNC(C(C=CCCC)O)=O)C2)nccc(NC)c1[N+](=O)[O-] C1(n2cc(CC(COC)O)nn2)CCCC(C(=O)NCCCC2CCOCC2)C1 CC(C)CC(CNC(=NCCc1ccnn1C)NC(c1ccsc1)C)CCO C1(C(=O)NCCC(C)N(C(c2nc(OC)nc(O)c2)=O)C)CCC2(CCC2)CO1 c1(C(=O)NC(CC2CN(C(CCC(=C)Cl)=O)C2)C)oc2ccc(C)cc2c1C C1(NC(C(CC)C)=O)CCCCC12CCN(C(c1ccn(C3CCCC3)n1)=O)C2 CC1(C(=O)NC2CCN(CCCO)C2)C=CCN1C(c1cc(C2CC2)[nH]n1)=O C1(NC(=O)COC2CCCCC2)CCCCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(CCC)(C)CC)=O)CCC2(C1)CN(C(C1(C)CCCCO1)=O)CCO2 N1(C(c2c(OC)scc2)C(=O)NCCC#N)CCCC(n2nc(C)cc2C)C1 N1(C(C(C)OCC#C)=O)CCN(C)C(CNC(C2(n3cccn3)CCC2)=O)C1 c1(N2CCC(OCCNC(C=C(C)Cl)=O)C2)cc(Cl)ncn1 c1(C(N2CC(CN(C)Cc3ccsc3Br)C2)=O)c(I)ccnc1F C1(C(N2C(CNC(N)=O)CCC2)=O)CCCCCCN1C(c1ccc(CO)o1)=O C(=O)(CC(C)(O)C(F)(F)F)NC1CC2CN(C(C(C)(C)CF)=O)CC1C2 Cn1ncc2c1CN(C(C1CCN1Cc1cccc3nonc13)=O)CC2 CCCC(CNC(=O)Cc1ncccc1F)C(=O)NCC(C)CN(C)C C1(NC(Cc2n(C)ncc2)=O)CN(C(C2(C)C=CCCC2)=O)CC2(CCC2)C1 CC1=C(C(=O)N2CCC2CNC(c2ccoc2C(C)C)=O)CCC1 N1(C(CCC2C(C)=NOC2=O)=O)CCCC(C)C1CNC(=O)C=C1CCN(C)C1 C1(C(=O)Nc2cc(C)ns2)COCCN1Cc1cncc(O)c1 Cc1cccc(C(=O)NC(C(=O)NCC(O)C(N)=O)C(C)(C)C)c1C c1(C(=O)NCCC(C)NC(C2CCC(CC)O2)=O)cc(C(F)(F)F)ccc1Cl C1(C(N2CC=C(C)C2)=O)CC2CCC(C1)N2C(C1(C(C)C)CC1)=O N1(C(C2(C#C)CC2)=O)CCCC(F)(C(N2CCC(O)(CC(C)C)C2)=O)C1 C1(CCC)(NC(c2nnn(C)n2)=O)CCCN(C(c2cccc(C(N)=O)n2)=O)C1 n12cc(cn1)C(=O)NC2C.C1(OCC(=O)NC2(CF)CC2)CC=CC1 C12(CCCN1C(=O)Cc1cccs1)CSCC(=O)NC2.N1(OC)CCC(C)C1 N1(C(C2(C)COCCO2)=O)CCC2C(C(=O)NCC(F)C3CCC3)C2C1 CCCC(C)(CC)C(=O)NCCCNC(c1ccc(C#N)c(C)c1)=O N1(C(=O)C2=CCCOC2)CC2CCC1CN2C(=O)Cc1cncc(Br)c1 c1(C(=O)NCCC(=C)CNC(=O)C(O)c2cnc[nH]2)cn2c(n1)CCC(C)C2 C1(CNC(c2ccc(COC)s2)=O)CCCCN1CCCS(C)(=O)=O N1(C(C2(N(C)C)CC2)=O)CCC(C2CCN(C(=O)C3=COCC3)C2)CC1 C1(C(=O)NC2CCN(C(C)(C)C)C2)CCC2(CCNCC2)O1 Cc1nc2cc(C(N3CCCN(C(C4(C(C)C)COC4)=O)CC3)=O)ccc2o1 C1(C(N(C)CCNC(C2(C(N3CCOCC3)=O)CCCC2)=O)=O)CCNC1=O C1(C(=O)Nc2cn(CC3CC3)nn2)CCCC2(CCC2)O1.C12COCCN(C1)C2 S(=O)(=O)(c1cnc(NCC2(S(C)=O)CC2)c(Cl)c1)N(C)Cc1cccc(F)c1F C(=O)(CC(C)(C)C(F)(F)F)N(CC(C)NC(Cn1c(C(C)C)nnn1)=O)C C=CCCC(C(=O)NCc1cc(O)cc(F)c1)NC(=O)CCc1ccco1 c1(N2CCCC(CNC(Cc3c(C)cco3)=O)CC2)ncc2ncn(C)c2n1 N1(C(C2(COC)CC2)=O)CCCC2(CCC(NC(=O)Cc3cc(C)[nH]n3)C2)C1 C1(NC(C2(C=C)CC2)=O)CC12CCN(C(=O)C(C)(C)N1CCCCC1)CC2 C1(N(C)C(c2ccc(Cl)o2)=O)C2CC3C(=O)OC1C3O2 N1(C(c2c(C)c(N)ccc2)=O)CCN(C(c2sc(Cl)cc2F)=O)C(C)CC1C c1(C(N2CC3C(NC(c4c(COC)scc4)=O)(C3)C2)=O)ccc2sccc2c1 c1(C(=O)NCC(CN(C(C(C)NC(N)=O)=O)C)(C)C)ccnc2[nH]ncc12 C(C(C(C)C(C)C)NC(c1c(Br)c(C)nn1C)=O)NC(CCC)=O C(=O)(C1Cc2ccccc21)NCC1(C(C)(C)O)CN(C(=O)CCc2cnoc2)C1 c1(C(=O)NC(C)C(C)NC(c2ccc3cncn3c2)=O)cccc2c1COCC2 C1(CC)CN(C(C23CC(CO)(C2)C3)=O)CCN1C(c1c(C)coc1C1CC1)=O c1(C(=O)OC)ccc(Oc2ccccc2)c(I)n1.C12(F)CN(C1)C(=O)CS2 N1(C(CC(=O)NCC)=O)CCCC1(C)CNC(c1cn(C2CCOC2)nc1C)=O C1(Cc2n(Cc3cnsc3)c(N3CCOCC3)nn2)CCC2(CC2)C1 c1(NC(C(N)=O)=O)cccc(NC(=O)C(O)Cc2cnc[nH]2)c1 Cc1cc(=NCCOCC2CCCCC2c2cccnc2)[nH]c(NCC2CC2)n1 c1(C(N(C2CCN(OC(=O)CC)CC2)COCC)=O)cc2c(O)cccc2[nH]1 C(N=c1[nH]c(=NC2CCCSC2)[nH]c2c1COCC2)c1n(C)cc(Cl)c1 N1(C(c2cc(C)c(CO)cn2)=O)CC(C)CN(C(=O)C=Cc2cocn2)CC1C S(=O)(=O)(c1c[nH]c(C(=O)N(CC(C)NC(=O)C(C)(C)C(N)=O)C)c1)NCCOC C(=O)(C(C)(C)C1CCN(C(C2CC(CF)C2)=O)C1)NCC(c1ccccn1)C Cn1ncc2cc(C(N3CC(NC(=O)C(C)(O)C4CCC4)CCC(O)C3)=O)sc12 C(=O)(C(C)n1cncn1)NCC1(C(C)NC(CC)=O)CC1 C1(NC(C(CO)OC)=O)CN(C(C2(C)CCOC2)=O)CC1CO CC(C)S(=O)(=O)C(C)C(=O)N1CCCC(N(C)C(c2ccn3ccnc3c2)=O)C1 C=CCC(C)C(=O)NCc1cn(C2CCN(C(=O)C(C)(C)C3CC3)CC2)nn1 C(C1C(=O)N1C)NC(C1CC1(C)C(F)F)=O.C=CC(C1CC1)SC.C(C#N)S c1(C(N2CC(c3ccccc3)(NC(C3C(C)CCO3)=O)C2)=O)occ2c1CCC2 c1(C(N(C(C)CN(C(=O)Cc2nc(=N)[nH][nH]2)C)C)=O)ncc(F)cn1 c1(C(N2CCCC(F)(C(N3CCCCC3CCO)=O)C2)=O)ncn2c1CCC2 N1(C(C(C=CC)O)=O)CCC(CNC(c2cn(C)nc2C(C)(C)C)=O)C12CC2 C1(CNC(CCS(N)(=O)=O)=O)CC2(CCN(C(=O)CCCC(=O)C3CC3)C2)CO1 C=C(C)CC(C(=O)N1CCSCC1C(=O)NC1CCC(C)CC1)OC C1(C(N(CCN(C(=O)CCc2cscn2)C)C)=O)CC1(F)F C1(C)(CC)C=C(C(=O)NC2CC3CN(C(=O)COCCc4ccccc4)CC23)C1 c1(C(=O)NCC2(O)CCCN(C(=O)CN3CCCCC3)C2)ccc(Br)c(CO)c1 C(=O)(CC(C)C(C)(C)NC(=O)CC(C1CC1)C1CC1)Nc1ccc(OC)nc1 c1(C(=O)OC)cc(CCC(=O)NCCN(C(=O)C(C)C2CCOC2)C)c[nH]1 C1(NC(C(=O)NC(C#C)C2CC2)=O)CNCCS(=O)(=O)C1 c1(OC)cc(C)cc(C(=O)NCC2(F)CCC(NC(=O)C(F)(F)C(C)O)C2)c1C c1(CN=C(NCC(CC)(C)OC)NC(C)COC)nc2cc(C)ccc2n1C Cc1c(F)cc(C(N2CCC(F)(C(=O)NCc3ccccc3)CC2)=O)cc1Br C=CCC(C(=O)OC1CC(C)OC(C)C1)C(C)C C1(C(=O)NC2CCC(N(C)C)C2)CC(O)CN1C(c1cnc(S)nc1)=O C1(CCC(=O)N(c2cn[nH]c2)CCOC)NC(=O)NC1=O CC1CCCC1(C)C(N1CC(O)(CN(C(=O)CC2(O)CCOC2)C)C1)=O N1(C(C2CC(NC(C(C)n3ccnn3)=O)C2)=O)CC2C(=O)NC(=O)C2C1 c1(C(=O)NC2CC(CCNC(COC)=O)C2)cc(C(F)(F)F)c(Cl)cn1 c1(CC)ccc(-c2nc(CCO)nn2-c2cnnn2C)cc1 N1(C(C(CC)OCC)=O)CCCC(C)(C)C1CNC(c1ccc2c(c1)COC2)=O C(CCCC(=O)NC1C=CC(C(=O)NCCCN(C)C(C)C)C1)SC Cc1ccc(NC(=O)C(N2CCC(c3cc(CCCOC)on3)CC2)=O)cc1C c1(NC(=O)NC(C)(C)C)cnc(O)cc1C(=O)OC1(c2cccc(F)c2N)CC1 C(CC(=O)NC(C)C(=O)NCC(F)CO)OCC O=C(CC(C1CC1)C1CC1)NCC1(C(=O)NCC2CCC(O)C2)CCCC1 CCC(C)(C)C(O)C(=O)N1CC(C=C)(CC(=O)Nc2cnc(C)c(C)c2)C1 c1(NC(C2CCCC(Nc3c(OC)cncn3)C2)=O)cn2ccccc2n1 Cc1nc(O)c(Br)cc1C(=O)NCC1CN(C(c2cncs2)=O)CC1C N1(C(c2cn3ccccc3n2)=O)CCOC2(CCN(C(C3CC4CC4C3)=O)C2)C1 N1(C(=O)C=Cc2ccco2)CCC(N2CCN(C(=O)CSC3CC3)CC2)CC1 C1(O)(C(C)NC(c2cc(C)ncc2)=O)CCN(C(=O)C(C)(C)CF)CC1 CCC(CC)C(F)C(=O)NCC(C)(C)CC1CN(C(=O)CC2CCN(C)CC2)C1 N1(C(c2c(-c3cc(C)on3)ocn2)=O)CC2CCC1C1CN(C3CC3)CC21 n1(CC(=O)NCC(O)CCNC(c2ccoc2Cl)=O)ncn2nccc2c1=O c1(OC)c(CNCC2(CC(N3CCCC3CO)=O)CCOC2)cccc1Cl c1(C(=O)NC(C)C(C)NC(=O)CCC2CC2(C)C)cnc2cc(Br)ccn12 c1(-c2ccc(NC(C(=O)NCC3CCCNC3=O)=O)cc2)ncc2c(n1)CCC2 Cc1c(C(=O)NC(CC(F)F)C(=O)NCC(C)C(C)C)cccc1C#N c1(N2CCC(C(C)NC(=O)Cc3cccn3C)CC2)cc(Cl)nc(S(C)(=O)=O)n1 Cc1ccc(COC(C)C(=O)NCC=CCNC(C2CCOC2(C)C)=O)cc1 CC1(C)CC(NC(c2csc(-c3ccoc3)n2)=O)CN1C(C1CC2(CC2)CO1)=O c1(CN(C(Cn2cc(CC(=O)OCC)nn2)=O)C2CC2)cccc(C(F)(F)F)c1 c1(C(=O)NC(CC)(CNC(=O)CC2(OC)CC2)CC)cc(C)c2c(c1)CCC2 Cc1c(Cl)c(C(=O)NCC(C2CCN(C(c3cnn(C)n3)=O)CC2)C)nn1C N1(C(C(C)N2CCC2)=O)CC(CNC(c2cc(N(C)C)nc(Cl)c2)=O)C(C)(C)C1 Cc1cc(Cl)nc(N)c1C(=O)NCCCCCNC(=O)CN(C)CCO Cc1cc(C)cc(S(=O)(=O)N2CCC(O)CC2C(N2CCOCC2C(C)C)=O)c1 C(=O)(C1CCCn2nccc21)NC1CC(C)(NC(C(CCC)NC(C)=O)=O)C1 C1(C(=O)OCC)CCCC(C(=O)NCC(O)CNC(c2conc2C(C)C)=O)C1 N1(CCOC)C(C)CN(CC(C)(C)COC2CC2)CC1C Cn1ccnc1CC(=O)NCC1CC1C(=O)NCCOCC1CCC1 C1(C(=O)NCc2ccc(Br)s2)CCN(Cc2cccnc2)C1=O C#CCCCCC(=O)N1CC(CNC(=O)C(C)Sc2ccc(N)cc2)(OC)C1 N1(C(CC=CC=C)=O)CC2CC(NC(C3CC34CCSCC4)=O)C(C2)C1 C1(C(N2CCC(CNC(C3(c4nc(C)[nH]n4)CC3)=O)CC2)=O)CC(=O)OC1(C)C Cc1nc(Br)c(C(c2nnnn2C)NCC2CCCC23CCC3)n1C C1(n2cnnn2)(C(=O)NCC2CCN(C(=O)CCc3ccco3)C2)CCOCC1 C=C(CC)CN=c1[nH]c(=NCc2cnc(O)[nH]2)[nH]c2ncn(C)c12 C1(NC(C(CC)CO)=O)CN(C(=O)CC2Cc3ccccc3N2)CCC1C C1(C(=O)NC2(CN(C)C(C3CC4CCC(C3)O4)=O)CC2)CCCCC12OCCO2 N1(Sc2nnnn2C2CC2)CCN(C(=O)CC2CC2)CC1.CC1C(=O)N(C)CC1 CCCC(C(O)C(=O)NCCC1CC=CCC1)NC(=O)COCCF c1(C(=O)NC2C=CC(CC(=O)Nc3cncnc3O)C2)cccc2ncccc12 c1(C(=O)NCC2OCCCN(C(C(=O)NCCOC)=O)C2)ccc(C#N)cc1F c1(CC)cc(C(N2CCCC(C(C)(O)CNC(=O)CN(C)CC)C2)=O)ccc1C C(=O)(CS(=O)CCC(F)(F)F)N1CCC(O)(CN(C(=O)Cc2ccccc2)C)C1 N1(CC(CSC)O)CCC2(CC1)CC2C(=O)N(CC(C)OC)C C(=O)(C1=NOC(CNC(=O)CNC(=O)OC)C1)N1CCC(N(C)C)(CC)C1 CC(F)(F)CCCC(=O)NC1CC(O)(CNC(c2ccc(C3CCC3)cc2)=O)C1 c1(-c2cn(C(CNC(C3CC(=C)C3)=O)C)nn2)cc(C)cc(F)c1 C(N=c1cc(C)[nH]c(=NCCc2cnn(C)c2)[nH]1)C1CC(OC)C12CCC2 CN1CC2CCC(C1)N2C(C1C2CCC(C2)C1NC(C1(C)CCCC1)=O)=O c1(C(=O)OC)ccc(N2CCCC(C(C)NC(=O)C=C(C)C(C)C)C2)nc1C N1(C(Cc2cccc(CC(C)C)c2)=O)CC(NC(=O)C=CC2CCCC2)C(C#N)C1 CC1(C)OCCC1CC(=O)NCCNC(C1C(C)(C)C1(F)F)=O CC1(C)COC(C)(C(N2CC(NC(C3CC(F)(CO)C3)=O)CC(F)C2)=O)CO1 Cc1coc(C(N2CCC(NC(c3ccc(-n4ccnc4C)nc3)=O)C2)=O)c1C c1(NC2C(SC)CC2)cc(-c2cc(-c3n(OC)ccn3)n[nH]2)c(F)cc1C C1(C(=O)NCC=CCNC(C(C)(C)CC2CCC2)=O)CC2CC(O)CC(C1)C2 c1(NC(c2n(CCCC)nnn2)C2(CCSC)CC2)cnc(C)c(Br)c1 c1(SC)c(C(=O)NC(C)CN(C)C(c2cnc(C(C)=O)s2)=O)cnn1C C1(C(=O)NC(CC(C)C)CNC(=O)C=Cc2ccccc2)CCCS(=O)(=O)C1 C1(CCNC(c2ccnnc2O)=O)CCN(C(c2ccnn2CC(F)F)=O)CC1 c1(OC)ncc(C(=O)NC(C2CN(C(c3ccc(N)cc3)=O)CCO2)C)cn1 C1(C(N(CCCOC)CCO)=O)CCCCN1C(=O)CCc1nc(C)no1 NC1CC(NC(C2(c3ccc(F)cc3F)CCCC2)=O)CCC1C(=O)O C1(CNC(CCC(C)N(C)C)=O)CCC(F)(CNC(C2CCO2)=O)CC1 C1(CC(=O)NCC2N(C(C(c3cscn3)N(C)C)=O)CC2)(N(C)C)CCCC1 CC1CCC(=CC(=O)N(CC(=O)NCC2(C(=O)N(C)C)CCCC2)C)CC1 C1(CC)C(NC(c2c[nH]nc2C)=O)CCN1C(c1ccn(CC)c1C)=O C=C=CCC(=O)NC(C)CN(C)C(c1cn(Cc2ccccc2)cn1)=O N1(C(C2N(CC)CCOC2)=O)CCCCC(CNC(c2ccc(Cl)s2)=O)C1 C1(COC(C)C(=O)NC2CC(C)(NC(C3CCC4CC34)=O)C2)CCCCO1 C1(NC(C2N(C(C(C)OCC#C)=O)CC(C)C2)=O)CC2C(O)C(O)CC12 C1(NC(c2ccnnc2S)=O)CC2CCCC(C1)N2C(=O)C(F)C1CCC1 N1(C(CN(C(C)C)C)=O)CC=C(CNC(C2CCC3CC3CC2)=O)CC1 O=S(=O)(c1nc(C(F)(F)F)cs1)N1CCn2nnc(Br)c2C1 C(=O)(C1=CCCC(C)(C)C1)NCC1CC(OC)CN1C(=O)Cn1cnccc1=O CC1CN(C(C2CCOC2)=O)CCCN1C(c1cc(C(F)(F)F)ccc1O)=O c1(NC(c2csc(-c3cnccn3)n2)=O)nccc2c(F)cccc12 CN1Cc2ccc(NC(=O)C(N3CCC(Cc4ccc(Cl)cc4)C3)=O)cc2C1 CC1(Oc2ccc(Br)cn2)CCCN(C(=O)Nc2cnn(C(=O)OC(C)(C)C)c2)C1 N1(C(C2C(C(C)C)(CC)C2)=O)CCCCC(N=c2[nH]nc(CO)s2)C1 c1(C(=O)OC)ccc(Cc2cnnn2CNCC(=O)NCCN(CC)CC)cc1 c1(C(N2CC(C)(NC(CCC3CCC(C)O3)=O)C2)=O)c(O)cccc1Cl c1(SC)cc(C(N2CC3CC2(CNC(=O)C2=CCSC2)C3)=O)ccc1[N+](=O)[O-] C1(NC(C2N(CC)CC2)=O)CCN(C(c2nscc2Br)=O)CC1 c1(C(=O)NCC2N(C(c3cn(CCC)nc3)=O)CC2)cccn(C)c1=O N1(C(=O)N(C2CCCC2)CCc2n(C)cnc2)CCCC2CC12 N1(C(CC2(C)CC2)=O)CC(NC(c2cccc[n+]2[O-])=O)CC2(CC2)C1 C(N=c1ccnc(NCC(c2ccsc2)C)[nH]1)c1c(CC)scn1 C1(C(N2CCN(CC(=O)NC(C)(C)C)CC2)=O)CCOC(=O)CC1 n1(CC(=O)NC(C2CN(C(C(CCCOC)C)=O)C2)C)ccc(=O)c([N+](=O)[O-])c1 c1(C(=O)NC2(C(=O)Nc3c(C)ccc(C)c3)CCSC2)ccc2c(c1)CCC2 N1(C(C(c2cccnc2)OC)=O)CC2CCC1C1CN(C(=O)C(C)(C)CF)CC21 c1(C(N2CCN(C(C(CC)c3ccccc3)=O)CC2CO)=O)nsc2ccccc12 Cn1nc2c(c1C(=O)NC1CC3CC1N(C(c1ccnnc1O)=O)C3)CSCC2 C1(C(N2C(C)CN(C(C3CC4(C3)CC4F)=O)CC2)=O)C2Cc3ccccc3C12 c1(C(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)ccncc1C(F)F CC1=NOC(C(=O)NC2CC(C(C)NC(c3cc(C)oc3C)=O)C2)C1C C1(CF)CN(CCC2CC=CC2)CC1C(F)F Cc1nc(C(C)C)sc1C(=O)N(C)CC1CCN(C(=O)C(C2(O)CCCC2)F)C1 c1(OC)cc(C(=O)N(C(C)CN(C)C(c2csc(C#N)c2)=O)C)ccc1Cl CN1CCCC(C(N2CC(C3CN(C(C4CC5C=CC4O5)=O)CCO3)C2)=O)C1 C1(C(=O)Nc2cc(Cl)c(I)cc2F)COC2(CCNCC2)C1 C1(NC(c2nc(CC)sc2)=O)CC(OC)CN(C(=O)C(O)CSC)C1 Cc1ccc(C)c(C(N2CC3(CO)CC2(C(=O)NCc2cccc(C)c2C)C3)=O)n1 c1(C(N(C)CC2N(C(C(F)=CC)=O)CCC2)=O)ccc(CCCN(C)C)nc1 C1(NC(c2cc(C)n(C3CC3)n2)=O)CN(C(c2cocn2)=O)CCC1C C#CCCCCCC(=O)NCC12CCCC1N(C(=O)C(C)(C=C)CCOC)CC2 Cc1cccn2ncc(C(N3CCC(C)(C)C3CNC(=O)Cn3nccn3)=O)c12 C1(CC(=O)NCCC(C)NC(=O)CCN(c2ccncc2)C)CCC(=O)NC1=O n1(CC)nc(C(=O)NCCN(C)C(C2CCCN2CC(C)C)=O)cc1O C(CCC(=O)Nc1nc[nH]n1)NC1(CSC)CC1 C1(NC(CNC(CCCC)=O)=O)CN(C(=O)C(c2ccccc2F)(C)C)CC1O c1(NC(C2N(c3cc(C#N)ncn3)C3C(C2)C3)=O)ccccc1S(=O)(=O)F N1(C(c2c(CC)n(C)cc2)=O)CCCC(C)(C(N2CCCCC2)=O)C1 N1(C(CSC(C)C)=O)CC2CN(C(=O)C(C)C(C)(C)C)CC2(C)C1 C1(C(=O)NC2CCN(C(C3CC(n4ccnn4)C3)=O)C2)C2CC3C(C2)C13 c1(C(=O)NC(C(C)NC(c2ncc(C)cn2)=O)CO)cnn2c1NCC(C)C2 C(=O)(C(C)CC(F)(F)F)N1C(CNC(c2c(Cl)nc(OC)s2)=O)CC1 N1(C(c2cccc(C)n2)=O)CCC(=O)NC2CN(C(=O)C(C)(Cl)Cl)CCC12 c1(C(N2CCC(CNC)CC2)=O)ccc2cnn(C)c2c1 C1(CNC(CC(=C=C)C)=O)CC2CCC1N(C(c1cncc3nc[nH]c13)=O)C2 Cn1[nH]c(C(N2CCCC2CNC(=O)CN2CC3CC3C2)=O)nc1=O c1(CC(N2CC(CNC(c3cnc(C(F)F)s3)=O)C(O)C2)=O)ccc(F)cc1F C1(NC(C(CCSC)O)=O)CC2(CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C1 C12(C(=O)OC)CCCC1(C(=O)N(CCCNC(c1cccc(C3CC3)c1)=O)C)C2 c1(C(N2CC3CC(NC(C4N=C(C)SC4)=O)C3C2)=O)cccc2c1NCCC2 c1(C(=O)NCC2N(C(c3ccco3)=O)CC2)ccccc1C(O)CF CC(C)C(O)C(F)(F)C(=O)NC1CN(C(c2ccoc2Br)=O)C2CCCCC12 c1(C(=O)OC)cc(NC(CCN(C(=O)C(C)(C)F)C)C(C)C)nc(Cl)n1 Cc1ncc(NC(=O)C(CC(F)F)N(C(=O)C(C)NC=O)C)cc1Cl C1(O)(CNC(c2nncs2)=O)CCCN(C(=O)COCc2cccnc2)CC1 C1(NC(C2C(C)=C2)=O)CC2CN(C(c3sccc3F)=O)CC12 C1(C(N(CCOCC=C)C)=O)N(C(=O)CCC(C)(C)C)CCC1(C)C c1(OC)cnc(Cl)nc1N1CCC(C)(NC(c2csc(C3CC3)n2)=O)CC1 CCC(C)(O)C(=O)NCCN(C(C12CCN(CC1)C2)=O)Cc1ccccc1 Nc1ccc(C(=O)NC2CC(O)CN(C(=O)Cc3ccno3)C2)nc1N C1(NC(CSCCN(C)C)=O)CN(C(=O)CC2CN3CCN2CC3)CC(C)(C)C1 C#CC1(CNC(=O)C(C)(CO)NC(=O)C(CC)N(C)C)CCOCC1 C1(CNC(C2C(COC)CC2)=O)CN(C(c2cc(F)ccc2C)=O)C2(CCC2)C1 Cc1cc(C(=O)NC2(C#N)CCN(Cc3cccnc3)C2)cc(Cl)n1 CC1CN(C(=O)Cc2cnoc2)CCC1CNC(C1(c2ncco2)CCC1)=O C12(C(=O)NC3(CO)C(C)CCCC3)CCC(CN(C(c3cc(=O)cc[nH]3)=O)C1)C2 C(C(CNC(C1CCOC(CC)C1)=O)S(C)(=O)=O)NC(c1cnc(CC)nc1)=O N1(C(Cn2nc(C)c(Cl)c2C)=O)CCCC12CCCSC2 N1(C(=O)CCc2ccc(Br)c(F)c2)CCOc2ccc(Cl)cc2C1 N1(C(C2(CCOCC)CCC2)=O)CC2CC(NC(=O)C(=Cc3c[nH]cn3)F)C2C1 C(CC(CC)C(=O)N(CCC(=O)NCC1COCC1O)CC1CC1)=CC N1(C(C(C(C)=O)(C)C)=O)CCC2(CC1)COC(CNC(=O)Cc1cccnc1)C2 C(N=c1[nH]c(=NCc2cccc(Cl)c2Br)[nH]c2cc[nH]c12)c1c(F)cccc1F N1(C(c2cnnc(C)c2C)=O)CC2CCCC2(C(N2CC(C)(C)CC2C)=O)C1 c1(C(N2C(CNC(C=CC)=O)CC2)=O)cnc2[nH]ncc2c1 c1(C(C)(C)NC(=O)C(O)Cc2ccncc2Br)nc2ccccc2s1 C(c1ccc(F)cc1)=CC(N1CC(NC(CCCc2ncc(C)o2)=O)C(C)C1)=O CC#CCCCC(=O)N(CC(C)N(C)C(C1CCCC(=O)O1)=O)C c1(-c2cc(C(=O)OC)ncc2)cc(C)c(S(=O)(=O)NCCCO)cc1C c1(C(=O)NCC2CCCCN(C(CC3C(C)C3(F)F)=O)C2)cccc2[nH]ncc12 N1(CCc2c(C)cccc2)C(=O)CN(CC)C1=O.c1(OC(F)(F)F)ccc(F)cc1 C[Si](C)(C)c1cccc(NC(C2(N)CC3(CCCCC3)C2)=O)c1 N1(C(C(C)N(C(=O)Cc2ccco2)C)=O)CCCC(F)(F)CC1 C(=O)(C(C)Cc1cccnc1)NCCC(C)NC(C1(C#N)CCC1)=O C(C)(C)(C(=O)NC1CC1)OC(C)C.C1(Cn2cc(C(C)(C)CO)nn2)COCC1 c1(C(N2C(Cn3cc(CN(C)S(N)(=O)=O)nn3)CCC2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(CC(C)CN(c2cccc(Cl)c2)C)=O)CCCC(C)(C(=O)N(C)CCO)C1 c1(C(C)NCc2ccc(C(=O)O)s2)ccc(Cl)c(Cl)c1 c1(CC(=O)NCC(CC)(C)NC(c2cnn(CCF)c2)=O)cccnc1O C1(C(=O)NC(c2ncc[nH]2)C)C2CCN(C(=O)C(C)CC3CCCC3)CC12 CC1CN(C(=O)NC2CCCN2S(=O)(=O)Cc2ccccc2)CC(C)(C)CO1 CCC(F)(F)CC(=O)N1CCC(CC(N2CCCC2(C)C(C)(C)C)=O)CC1 c1(CCC(=O)NC(C(C)NC(C2C(F)(F)C23CC3)=O)(C)C)ccccc1[N+](=O)[O-] C1(CC)CCC(C)N(C(=O)CC(C)(C)N(C)C(C2(C(N)=O)CCC2)=O)C1 c1(NC(C(C2CCN(S(=O)(=O)c3nccs3)CC2)C)=O)cnc(Cl)c(C#N)c1 N(C(=NCC1COC(C)(C)C1)NCc1ccccc1)CC1(OC(C)C)CCCC1 c1(C(=O)NCCC(CNC(C2C(=C)C2)=O)O)nc(O)nc(O)c1OC C1(c2nnnn2C)(NC(c2ccc(OCCC)cc2)C(C)C)CC12CCOCC2 c1(C(N(C2CCN(C(C3CCC(C)O3)=O)C2)CC)=O)c(C)nc2sccn12 n1(CC)nc(C(N2CC(NC(C3(c4ccc(Cl)cc4)CCC3)=O)C2)=O)ccc1=O c1(NC(c2nc(C(N)=O)sc2)=O)ncc(Cl)nc1Cl.c12ccc(Cl)cc1NC2=O N1(C(C(C)C)=O)CC2CCCC2(CNC(=O)C(C)Cc2cccnc2)C1 C(=O)(C1CCc2ccccc21)N1C(CNC(=O)CCCCO)CC(F)C1 Cc1ccc(C(=O)NC2CC3(C2)CN(C(C2CC4C=CC2O4)=O)C3)cc1[N+](=O)[O-] C(CCCC(C)(F)F)NC(C(C)N(C)C(c1ccc(N(C)C)cn1)=O)=O C1(NC(c2cc(C(C)=O)oc2)=O)CC(NC(=O)C(C)C2CC2)CC1O C(C(COC)CC(=O)N1CCC(CO)(CNC(=O)CC(C)C2CC2)CC1)OC N1(C(=O)OC)CCN(N2CCC(N3CC(C)OC(C)C3)C2)CC1 c1(C2(OC(C)(C)Cc3ccc(=O)n(C4CCCC4)c3)CCOC(=O)CC2)cc(C#N)ccn1 n1(CC)cnc2c(N(C)CCOC(C)COC)[nH]c(=NCC(C)S(N)(=O)=O)nc12 C1(C2CCN(C)CC2)(C(N(C2CC(NC(c3c(OC)cccn3)=O)C2)C)=O)CC1 c1(C(N2CCC(NC(=O)C=CCO)CC2C2CC2)=O)cc2ccccc2cc1F CN1N=C(CC(=O)N2CC(NC(c3ccc(O)nn3)=O)CC23CCCC3)CC1=O c1(C(=O)NC2CC(CNC(c3nocc3C3CC3)=O)C2)ccc(Br)cn1 CC1(NC(=O)CCOC2CCC2)CCN(C(c2ccccc2C(F)(F)F)=O)CC1 C=CC1(CC(=O)NC2CN(C(c3cc(CC)no3)=O)CC2SC)CCOCC1 CS(=O)(=O)c1ccc(OCC2CCC3(CN(C(=O)C(O)CCl)C3)O2)cc1 c1(CC)ccc(Cl)c(C(=O)NC2CN(C(c3cccc(C)c3)=O)CC2C)c1 Cn1nc(Br)cc1C(N1CC(CNC(c2cn(CCF)nn2)=O)C(O)C1)=O CCCCCCCCCC(=O)NC1CCN(C(c2csc(C(C)=O)n2)=O)CC1O C=CC(CC)CC(=O)N1CCC(C(=O)Nc2nc(C3CC3)c(Br)s2)C1 c1(CC#N)cccc(C(=O)NC2CC(NC(c3cc(Cl)c(Cl)s3)=O)C2)c1 CCC(C)(CCC(C)C)C(=O)N1CC(F)(CNC(=O)CN2CC(C)(C)C2)C1 CC1CCC(O)CN1C(C1(NC(c2cc(C(N)=O)[nH]n2)=O)CC(F)(F)C1)=O CC1CN(C(c2ncncc2F)=O)CC1NC(c1cn(C(C)(C)C)cn1)=O CC1(C)CCN(C(c2ccc(F)o2)=O)CC1CNC(=O)CC1CC1C(F)(F)F C1(C)(CNC(C(c2ccc(Cl)cc2)C)=O)CC(F)(F)CN1C(=O)CC(F)F CC(CCN=c1nc2ncccc2c[nH]1)NC(C1(O)CCSCC1)=O c1(SC)cccc(C(=O)NC2CCCN(C(=O)Cc3cc(C)nn3C)C2)c1Cl c1(C(=O)NC2(CNC(c3n(CC)ncc3)=O)CC2)cn(C(C)C)nc1Br C1(CCOC)CN(C(C2CN(C)C(=O)N2)=O)CCN1C(=O)CN1CC2CC2C1 c1(C(=O)NC(C)CCNC(c2cc3n(c2)CCOC3)=O)cnn2c(N)ccnc12 N1(C(CCN(C)CCO)=O)CCC2(CC1)CC2C(=O)Nc1cncc(C#N)c1 N1(C(c2c(Br)cn(C(C)C)n2)=O)CCc2c(CCN(C)C)cccc2C1 Cc1ncc(C(=O)NC(C)CN(C(=O)CCc2csc(=N)[nH]2)C)c(C2CC2)n1 N1(C(C(CC)N(C)C)=O)CC2CC(NC(c3cncc(C(C)C)c3)=O)CC(C2)C1 C=C1CCC(C(N2CCC(C(=O)N(C3(CC)CC3)C)(CC)C2)=O)CC1 c1(C(c2nnnn2CCCOC)NCC2(CC)CCCO2)c(C)noc1Cl C(=O)(CC(C)(O)COC)NC1C(NC(c2c(C(=O)OC)cco2)=O)CCCC1 C(=O)(CCS(C)=O)N(C1CC(C(=O)NCC2(n3nccn3)CC2)C1)C c1(C(=O)NCCCC#C)ccc2c(c1)CN(C(c1ccoc1)=O)CC2 C1(CNC(C2(CC=C)CCOC2)=O)CC(C)(C)CN1C(=O)C1=C(C)CCC1 N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(c2cc(C)ccc2O)=O)CC1C C1(CCC)CN(C(c2cnc(C)nc2)=O)CCN1C(c1nnn(C(C)(C)C)n1)=O N1(C(C(CCCNC(CCN(CCC)C)=O)O)=O)CCC2(CNC(=O)O2)C1 C(C(F)(F)C(=O)NC(C1CCN(C(c2cc(C)nn2C2CCC2)=O)C1)C)OC C=C(Cl)CCC(=O)NC1CN(C(C2C=C(C)CS2)=O)C1 c1(CNCc2c(COC)cccn2)ccc(C)cc1OC1CCOCC1 C1(NC(Cn2nc(C)oc2=O)=O)C2CC3CN(C(C4CCCCS4)=O)C1C3C2 N1(C(CC=CCC)=O)CC2CCCC(NC(c3cnc4ccnn4c3)=O)(C2)C1 c1(C(=O)NCC2(CCNC(C(C(C)O)N(C)C)=O)CC2)sc(C#N)cc1Cl c1(C(=O)NC2CN(C(CCCOCC)=O)C(C)C2)cc(C)ccc1C1CC1 Cn1c2c(ccc1=O)C(NC(=O)NCCc1nc(C(F)(F)F)n[nH]1)CCC2 O([Si](C)(C)C(C)(C)C)C(C)CNc1ccc(Cl)cc1Cl C1(CNC(CS(=O)(=O)NCC)=O)CC2(CCC2)CN1C(c1c(Cl)cnn1C)=O N1(C(CCCNC(=O)OC)=O)CCC2CN(C(C3(SC)CC3)=O)CCC2C1 Cc1ccn2ncc(C(N3CCN(C(C4CSc5ccccc5O4)=O)CC3)=O)c2c1 N1(C(c2c(Cl)sc(C)c2C)=O)CC2CCCC(N(C)C(C3CC3F)=O)C2C1 N1(C(CCC(=C)C)=O)CCC(C)C(CNC(c2ccc(N)c(SC)c2)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)N(C1CCN(C(c2nc(C(=O)OC)sc2)=O)C1)C c1(SCC(N2CCC(NC(c3ccn(C(C)C)n3)=O)CC2)=O)ccc(F)c(F)c1 N1(C(CCCCCSC)=O)CCC(C2CC2NC(=O)C(C)(C2CC2)OC)CC1 Cc1ccc(S(=O)(=O)N2CCOCC2CC(=O)Nc2ccc(O)cn2)c(F)c1 N1(C(C2(CC#C)CCCC2)=O)CCCC(C)(CNC(=O)CC(C)(O)C2CC2)C1 C1(NC(C23CC(C)C2C3)=O)CN(C(=O)C(c2ccccc2)=O)C2(CCOCC2)C1 N1(C(C(C)SCc2ccccc2)=O)CC(NC(c2csc(CO)n2)=O)CC(O)C1 c1(C(=O)NCC(CN(C(c2c(C)oc(Cl)n2)=O)C)C)ccc2sccc2c1 C1(NC(C=CCCC=C(C)C)=O)CN(C(C2(CO)CC2)=O)CCC1CO Cc1nc(-c2cccnc2)[nH]c1C(=O)NC(C)(CNC(C1CC12CC2)=O)C(C)C C1(NC(CCN(CCC)C)=O)(CC)CCCN(C(C2(C#N)CC2(C)C)=O)C1 C1(C(=O)NCC(C)(C)C2CC2)CC(CC)C1 c1(Cc2cc(C(=O)NC3CCN(C(C)=O)C3C)n(C)n2)ccc(Cl)cc1F Cc1cc(F)ccc1C(O)C(=O)NC1CC(NC(=O)Cc2cnns2)C1 C1(CC=C)(NC(c2cccc(CNC(=O)CN3CSCC3=O)n2)=O)CCCCC1 C1(C(=O)NC(CCNC(CNC(=O)OC)=O)C)CCCN1C1CCCCC1 CCCCC(C)C(=O)N1CCC(C)C(CNC(c2cnc(O)cc2C)=O)C1 Cn1nc(C(=O)NCCC2(O)CN(C(c3c[nH]nc3C(F)F)=O)C2)cc1O C(=O)(CCCC(=O)N(C1CCC(NC(=O)C=CCOCCOC)CC1)C)OCC Cc1onc(C(=O)NC2CN(Cc3ccnc(F)c3)CC2F)c1C c1(C(=O)NC2CCCN(C(C(=O)NCC)=O)C2CC)ccc2cnn(C)c2c1 c1(CC(=O)NC)cccc(NC(=O)NCC(N2CC=CC2)C)c1 C(CN=c1[nH]cc2ncnc-2[nH]1)c1c(C)non1 C(=O)(CCCOC(N(C(C)COC(C)(C)C)C)=O)NC(C)(C)C C(CCCC=C)(C(=O)NC(CO)CC#C)NC(C(CC#C)O)=O C1(CNC(c2cc(CCC)n(C)n2)=O)CC2CN(C(=O)C=Cc3cscn3)CC12 C(=O)(CCN=[N+]=[N-])N(C1CCCC1)CC(=O)NC(c1cccs1)CC CCC(CC)(CC(=O)OC)C(=O)N1CC2CC3CC2C1C3C(=O)O C1(C)(CNC(C(C(C)C)O)=O)CN(C(=O)CCc2cc(Cl)no2)CCO1 C1(CCC(=O)OC)CCC(NC(=O)CN2CCCC2)C1.C12CCN1C2=O N1(C(c2c(Cl)cnc(C)n2)=O)CC(NC(c2cn(C)cc2C)=O)C2(CCCC2)C1 C1(c2nnnn2CC(C)(CC)N(C)C)(NCCCCCC)CC2CCC(C1)S2 C1(CNCCC(=O)OCC)CCc2ccccc2C1.C12(CCC1)CC(=O)N2 c1(C(=O)NCC2CN(C(CN(C(=O)OCC)C)=O)C(C)C2)c(N)ccc(F)c1C N1(C(C(CC(C)=O)C)=O)CCC2C(CCCN2C(c2coc(Cl)n2)=O)C1 c1(CN2CC(CNC(CCOCC)=O)OCC2)ccc(F)cc1F C1(C(N2C(CN(C(=O)CCC3CC3)C)CCC2)=O)CC2CCC1CC21OCCO1 C(=O)(CC1OCc2ccccc21)NCCOC1CN(C(C(C)C(C)C(C)(C)C)=O)C1 c1(C(=O)NNC(c2ccc3c(n2)CCCC3)=O)ccc2cc(Cl)ccc2c1 C(=O)(C(F)(F)C(F)F)NC1CC(CNC(Cn2nc(C)c(Cl)c2)=O)C1 O=C1NCC2(CO1)CN(C(C1CC(n3cc(C(N4CCCC4)C4CC4)nn3)C1)=O)C2 N1(C(c2c(CC)onc2C)=O)CCC2C(CCCN2C2CC2)C1 C(=O)(C(CCCC(C)C)N1CCCC1Cc1cnn(C)c1)NCCC C1(C(=O)NC2C(C)CN(C(C3(F)C(C)(C)C3(C)C)=O)C2)CC1C1CC(F)(F)C1 N1(C(CC(C)C2CCCCC2)=O)CCN(C(=O)C(F)Cc2ccccc2)CC1 C(=O)(C(CCC)C(=O)OC)NC1C(C(=O)NC(c2cnn(C)c2)C#C)CC1 c1(C(=O)NCC(CC)NC(=O)C(C2CC2)OC)cnc(O)c(C(C)=NO)c1 N#Cc1cccc(NC(C2CCCCC2NCc2ccccc2CO)=O)c1Cl c1(N2CCC(CSC)C2)nc(-c2ccccc2)nc(=NC(C)Cn2ccnc2)[nH]1 n1(C(C=C)C)nc(-c2cnn(CCO)c2)nc1C1CCCOC1 CC1CN(C(=O)C(=O)Nc2ccc(CN3CCOCC3)cc2)C(C)(C)C1 C1(CNC(c2cc(C)n(C(C)(C)C)n2)=O)CN(C(=O)CC2CC=CC2)CCCO1 C1(NC(CCc2ccn(C)n2)=O)CCCCC1CNC(=O)CC1CCCCC1O C(=O)(C(C(C)O)N(C)C)NCc1c(C(N(CC(C)C)CC(F)F)=O)n[nH]c1 Cc1nc(C)n(CC(=O)NCC2CCN(C(c3ccc(CC(C)C)nc3)=O)C2)n1 C(CCCC(=O)N(C)CCNC(C1CC2(CC2)C1)=O)OCCC=C CC(CN=CCc1ccccc1)NCC1CCC(C)(C)C1 CC1=C(C(=O)N2CCN(C(c3cncc(Br)c3C)=O)CC2C)C(=O)OC1(C)C C1(NC(c2cnn(CCC)c2C)=O)(CNC(=O)C2=CCCC2)CC2CCC1CC2 c1(OC)ccc(C(N2CCCC2CN(C)C(c2ccsc2OC)=O)=O)cc1F N1(C(C2CN(C(=O)OC(C)(C)C)C2)=O)CC2CC3CC(C2)CC1C3.OC C1(C(N2CC3(C(NC(C4=CC(C)(C)C4)=O)CCC3)C2)=O)CNC2=C1CCCC2 C1(C(=O)NCC2(CNC(=O)CC3CC(F)C3)CCC2)CCC(=C2CCC2)CC1 N1(C(CC(=C)C)=O)CCCC2C(NC(C3CC4(CSC4)C3)=O)C(C)(C)C12 C1(NC(C2CCC(F)C2)=O)CC2(CCN(C(=O)CCc3ccc(F)cc3Cl)C2)C1 c1(C(N(CC(CC)NC(=O)CCn2ccnn2)C)=O)coc(C2CCC2)n1 C(=O)(CCC1CCc2ccccc21)NCC1(C)CCCN1C(=O)CNS(N)(=O)=O Cc1cc(F)c(NC(C2CCCN2C(c2ccccc2CO)=O)=O)cc1[N+](=O)[O-] N1(C(C2CC(=O)NC2)=O)CC(C2CN(C(=O)CC3CCNC(=O)C3)C2)C1 Cc1ncc(Cl)cc1NC(C1(NC(=O)Cc2cncn2C)CCN(C)C1)=O CC1CN(C(C2(CO)CC2)=O)CC(CCNC(c2n[nH]cc2Cl)=O)O1 Cc1c(C(=O)NCc2ncccc2CNC(=O)C(C(C)O)N(C)C)cnn1C c1(C(N(C2CCN(C(C3CC(C)N(C)C3)=O)CC2)C)=O)ccc(F)c2ccsc12 C(=O)(CCCC(F)(F)C(F)(F)F)N1CC2(N(C(CC(CC)OC)=O)CC2)C1 c1(C(C(=O)NCC2N(C(CCCCOC)=O)CCC2)C)ccc(C)c(Br)c1 C(N=C(NCCF)NC(C)(C)C(=O)NC)C1(CCC)CC1 c1(NC(C2CCCCCC2)(c2n(C(C)C)nnn2)CC)cnnc(S(C)(=O)=O)c1 CCC(CC)CCC(=O)NC(CC)CC(=O)N(CCCN1CCCC1)C c1(C(=O)NCC(CC=C)NC(=O)C(C)OC)ncc(C2CC2)cc1F C(C(CNC(c1cccc(C(C)(C)C)n1)=O)C(F)(F)F)NC(C(CC=C)C)=O c1(C(N2CC(N(C)C(c3cc(Cl)cn3C)=O)C(F)C2)=O)cc2n(c1)CCC2 c1(C(=O)NC2CC(F)(CNC(c3c(CC)noc3C)=O)C2)cc([N+](=O)[O-])oc1C c1(C(C)(C)C)cccc(C(=O)NC2(C)CC(NC(C3CCC(O)C3)=O)C2)n1 C1(NC(=O)OC(C)(C)C)C(C2CC2)CCN(N2CC3CC(O)CC3C2)C1 C1(CN(C)CCC2CCC2)CCCCN1CCSC(F)F N1(C(c2csc(C)c2C)=O)CC2(CCN(C(=O)C(C)(C)c3cnco3)C2)C1 C1(N(C(CC(C)NC2CC2)=O)CC2CC2)CCN(C(=O)C2=CCSC2)CC1 c1ccccc1C.CCC(C)(c1nnnn1C(C)C)NCCC(C)COC C(CCCC(=O)NC1(C(N2CCC(NC(C)=O)C2)=O)CC(O)C1)SC C(=O)(N=c1cc[nH]c(C2CCC2)c1)C1N(Cc2cc(C#N)cc(Cl)c2)CCSC1 c1(C(N2CCC(OCc3ccccc3)C2)=O)cccc(Br)c1Br c1(C(N2CCOCC2CC2CCC2)C(=O)NCCC#N)cccc2c1nnn2C c1(NC(C(c2ccc(F)cc2)(C)OC)=O)cc([N+](=O)[O-])ccc1C#N C(=O)(C(CCOCCO)NC(=O)Cc1cnsc1)N(C)CCN1CCCCC1 CC(C)CC(CC(=O)NC1COCCOC1)NC(c1cccn1C1CC1)=O Cc1sc(O)nc1C(=O)NC1CC(C(=O)NC(C)CCC(C)C)C1 C(CCC(C)C(=O)N1CC(CNC(c2ccc(C)c(C)c2)=O)C(F)(F)C1)OC C1(C(=O)NCC(CO)NC(C2CC(=C3CCC3)C2)=O)(OC)CCC1 c1(OC)ccc(F)c(C(=O)NC(CNC(c2cc(Cl)cc(Cl)c2)=O)CO)c1N C(CCC(O)C(=O)Nc1cccc(Cl)c1)NC(c1cnn(C)c1Cl)=O C1(O)(CNC(C2(OCC)CCCC2)=O)CCN(C(c2scnc2C(F)F)=O)C1 C12(C(=O)NCC(c3ccc(F)cc3F)NC(CSCC#C)=O)CC1COC2(C)C N1(C(C2N(CC)CC2)=O)CC(C)CC1C(=O)NCCC1(COC)CC1 CC1CN(C(c2cccc(O)n2)=O)CCC1CNC(=O)CC(C)(C)C1CC1 C1(C(=O)NCC(C=C)(C)C)C(CC)CCN1C(=O)C(C1CC1)OCC C1(c2ccccc2)(CC)CCCC(=O)N1.N12C(CCCC1C)CNC2=O C(=O)(CC1=CCN(C)CC1)NC1CN(C(C=C(COC)C)=O)C(C)CC1 N1(C(c2ccccc2Br)=O)CC2CCC1CN2C(C1(CO)CC1)=O c1(OC)cc(C(=O)NC2(C)CCCN(C(c3ccc(C)nc3)=O)C2)cc(Br)c1 NS(=O)(=O)CC(=O)NCC1CN(C(c2csc(-c3ccoc3)n2)=O)CCO1 n1(CC)cc(C(=O)NCC2CC2CNC(c2cocc2Br)=O)c(C(C)C)n1 c1(C(N2CC(C(F)(F)F)OC(C)C2)C(=O)NCC)c(F)cc(Br)cc1F c1(OCC)ccc(S(=O)(=O)N2CCOCC2)cc1C(=O)NC1CC2CCCCCC12 C1(NC(CC2(C)CCS(=O)(=O)N2)=O)CC2CCC(C1)N2C(=O)C(F)(F)C1CC1 c1(C(=O)NCCC2CCC(NC(C3CCC=CCC3)=O)C2)ccnn2ccnc12 C1(C(C)C)CN(C(c2cc[nH]c2)=O)CCN1C(c1ccc(-c2cnccn2)s1)=O c1(CC(=O)NC(C2(CNC(c3[nH]cc(CC)c3)=O)CC2)C)ccnc(F)c1F CCCC(F)(F)C(=O)NC(C)C(C)C(=O)Nc1cncc(F)c1 c1(C(N2C(CN(C(=O)Cc3cc[nH]n3)C)CCC2)=O)cc(N)ccc1F CC(C)CCCCC(=O)N1CC2(CO)CC1(C(=O)NCC1(O)CC1)C2 c1(CC(C(=O)NC2(C)CC(NC(C3(CO)CCCO3)=O)C2)O)ccc(F)cc1 c1(N2CC(O)(CCNC(c3c(C(C)(C)C)ocn3)=O)C2)ncnc2c1CCO2 C1(NC(=O)CCNC(c2ccccn2)=O)CN(C(=O)C#CC2CC2)CC12CC2 c1(NC(C(C(C)C)NC)=O)cccc(C#CCO)c1.C12CCCN(C1)C2=O C1(SC)CN(C(c2ccccc2)C2CC2F)CC1n1cc(CCCC#N)nn1 c1(C(=O)NC(C)CCN(C)C(C2CCCCS2)=O)cccc2ccsc12 c1(C(=O)NC2CCCC(NC(c3cnc(O)c(F)c3)=O)C2)csc([N+](=O)[O-])c1 C1(C)(NC(=O)CCO)CN2CCC1CC2.c1(C(C)OC2COC2)nocc1C=O C=CCCCCC(=O)NCCC1C(C)CCCN1C(c1cc([N+](=O)[O-])n[nH]1)=O C1(C(=O)NCC(C)(C)CNC(=O)CCCc2nccs2)CC(C2CC2)C1 C1(C(N(CCOCCN(C(c2csc(C)c2C)=O)C)C)=O)CC(C)OC(C)C1 C1(C(CNC(=O)C(c2ccccc2)F)F)CCN(C(=O)C2=CSCS2)CC1 Cc1cc(N)c(C(=O)NCc2ccc3nn[nH]c3c2)c(F)c1 C=CC(C)(O)CC(=O)NCC(C)(CNC(c1sc(C2CC2)nc1C)=O)OC c1(C(=O)NC2CCCN(C(=O)COc3ccccc3O)C2)c(F)cc(Br)cc1Cl C(=O)(C(C)N(OC)C(=O)C1CCC1NC(=O)CCc1nc(C)no1)OC CC(C)(O)C(F)(F)C(=O)NC1COC2CN(C(C3CC3C(F)F)=O)CC12 N1(C(c2n(CC)ncn2)=O)CC(NC(=O)CC2C=CS(=O)(=O)C2)C(C2CC2)C1 C1(C(CC)NC(c2ccc(-n3cccn3)cc2C)=O)CN(C)CC(C)O1 CN=c1[nH]cc(C(N2CC(NC(=O)C=CC(c3ccccc3)=O)C(O)C2)=O)o1 C1(CC(=O)NCC(F)F)CCCC(NC(=O)CC2CCOCC2)C1 C1(NC(C(N2C(C)(c3cccc(C(N)=O)c3)CCC2)=O)=O)OCC2CCCCC12 c1(-c2nc(CCOc3ccc(CCC)cc3)on2)ccc(-c2cccs2)cc1F N1(CCNC(C2CC(SC)C2)=O)CCN(C(=O)C(C)OC2CC2)CC1 C1(NC(C2CC2C(F)F)=O)CCC2(CC1)CN(C(C1CC13CCCC3)=O)CCO2 N1(C(Cc2cc(-c3nc(C)sc3)sc2)=O)CCCC(N(C)C(C2CC(F)C2)=O)C1 CC(C)C(C(=O)NCC1(CNC(C2C(Cl)(Cl)C23CC3)=O)CC1)n1cnnc1 C1(CNC(C2(C)C=CCCC2)=O)CCCCCN1C(c1ccc[nH]1)=O c1(C(C)=O)cc([N+](=O)[O-])ccc1NC1CC(C(=O)NC2CC23CCOCC3)C1 c1(OC)cnc(F)c(C(=O)NCCCC(C)NC(=O)C(C)(C(C)C)OC)c1 C1(C(=O)NC2CCC(C)(C)C2)CN(C(c2ccncc2F)=O)C2(CCC2)C1 c1(C(=O)NC2CC3CN(C(C=CCCC(C)C)=O)C2C3)ccn2ncnc2c1 c1(OCC)nc(NCC2CN(C(=O)CCC3CC3)CCO2)ncc1C N1(C(c2c(CCC)cccc2)=O)CCCC(NC(C2CCC(C)(C)O2)=O)C1C N1(C(CNC(CNC(C)=O)=O)=O)CC(NC(c2ccc(C)nn2)=O)C(F)C1 c1(C(C(=O)NCC(=C)C)N(CCCCSC)C)cc2ccnc(Cl)c2s1 C1(NC(c2nc(Cl)ccc2F)=O)CN(C(c2ccns2)=O)CC1C1CC1 C1(O)(CNC(c2ccc(C(N)=O)[nH]2)=O)CCN(C(C2CCCC2C2CC2)=O)CC1 C(CCC(F)(F)F)(C(=O)N1CCCC1C1CC1)CNC(=O)CCN1CCCC1 C12(C(=O)NC3(CNC(C(C(C)(C)C)O)=O)CCOC3)CCC(C(C)=O)(CC1)CC2 c1(C(=O)NC(CCNC(C2(OC)CC2)=O)C)cc(Cl)cc(Cl)c1[N+](=O)[O-] N1(C(c2c(SC)ccc(N)c2)=O)CCN(C(=O)COc2ccn(C)n2)C(C)C1C C1(C(=O)NCC2(C)CCN(C(=O)CCc3nncnc3O)C2)(OCC)CCSCC1 C(CCCCC(=O)N1CCC(C(C)NC(=O)CCc2csc(=N)[nH]2)C1)OC C1(NC2(C)CNC(=O)C2)CCNCCC1c1ccccc1 c1(CN2C(C)(C(=O)Nc3cccc(NC(=O)OC)c3)CC2)cc(F)c(F)c(F)c1 c1(OC)ncc(C(N2CCCS(=O)c3ccccc32)=O)c2ccccc12 C(CC1CC1)(C(=O)NCC(O)CCNC(c1csc(CCP(C)(C)=O)n1)=O)OC Cc1cc(Cl)cc(Br)c1NC(C1CCN1C(c1cc(Br)cc(Cl)c1F)=O)=O C1(NC(C2(COC)CCC2)=O)CC2(CCN(C(=O)CN3C(=O)CCC3=O)C2)C1 C(C)(C)(CC(F)C(=O)NCCOC(=O)C1CC1)NC(C1C(C)CC(=O)CC1)=O N1(C(C(COC)OC)=O)CCN(C(c2cc(OC)ncn2)=O)CC(O)C1 Cc1ccc(N)c(C(=O)NCC2(NC(C3CCCC3O)=O)CCCCC2)c1 C1(COC)CC(C(=O)NCCC(C)c2cn[nH]c2)N(C(=O)CCc2cn[nH]c2)C1 N1(C(c2c(OC)scc2)=O)C(CNC(c2cnn(C)c2OC)=O)CC2COCC12 N1(C(C(C)C)=O)CCN(C2CCN(C(c3cccc(O)n3)=O)CC2)CC1 c1(OC)ccc(Cl)cc1C(=O)NC1CC2(C1)CC2NC(c1[nH]c(C)nc1C)=O CCC(CC(=O)N1CC(CC(C)NC(=O)Cc2sc(S)nc2C)C1)SC N1(C(C=CC(=O)NC2CC2)=O)CCC(C2CCN(C(=O)Nc3ccccc3)C2)C1 c1(C(N2CC(CNC(CCCOC)=O)C(C(F)(F)F)C2)=O)ccnc(Cl)c1N c1(C(=O)NCCCC2CN(C(=O)CCC3CCC3)CCO2)c[nH]nc1[N+](=O)[O-] CC1=C(C(=O)NC2(C)CCCN(C(c3cscn3)=O)C2)S(=O)(=O)CCO1 c1(OC)cccc(C(N2CC(C(O)C(=O)NC3CC4C=CC3C4)C2)=O)c1 Cc1ccc(C(C)NC(C2CC(NCc3cnccc3Cl)C2)=O)cc1F C1(CC(=O)N(C2CCN(C(c3cc(C)n(CC)n3)=O)C2)CC)CC2CCC1C2 CCC(CCC(=O)OCc1cn(CCNC(c2ccc(Cl)cc2NC)=O)nn1)OC CCCC(C(=O)N(CC(C)C(=O)NC1CC1)CCO)OC C1(C(=O)NC(c2ccncn2)(C)C)CCCN(C(=O)C=C2CCCCC2)C1 CC1CCC(C(=O)NCC23CC(CN2C(=O)CC2CCC24CCC4)C3)CC1 C1(N(C(c2n(C(C)C)ccc2)=O)C)CN(C(C2CC3(CCCO3)C2)=O)CC12CC2 CN(C1C(=O)Nc2ccc(F)cc21)CC1Cc2ccccc2CN1C(=O)NC CC(O)(C(=O)N1CC(OCCC#CCO)C1)C1CCCCC1 C1(OC)CC(NC(=O)CCc2ccoc2)CN(C(c2coc(C(F)(F)F)c2)=O)C1 c1(C(N2CCC(C(=O)Nc3n(CC)nnn3)C2)=O)cc2c(s1)CCC2 C(CC(C)N=c1[nH]c(N2CCCCCCCC2)nc2ncn(C)c12)SC C=CCC(C(=O)N1CC(C(N2CC(C)(COC)C2)=O)C(C=CC)C1)C(C)C Cc1cocc1C(=O)NCC12CC(NC(=O)C(C3CCCCC3)=O)(C1)C2 C12(SC)CCC(CC1n1cc(-c3ccc(C(=O)NCC4CC4)cc3)nn1)C2 c1(C(=O)NCc2nccnc2Cl)c(O)c(Cl)cc(Cl)c1Cl.C12CCCN(C1)C2=O S(=O)(=O)(c1cccs1)NC1CCN(CC(=O)Nc2cc(OC)ncc2)CC1 C#CC1CCCCN1C(C1(C)CN(C(=O)CC2CCC(C)(C)O2)CC1C)=O C(C(C)(C)C1=CCCCC1)NCCC(c1cc(Br)c(OC(F)F)nc1Cl)c1n(C)nnn1 N1(C(CNC(=O)OC)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1CCC12CCC2 CN=c1[nH]c(=NC(C)c2nccc(=N)[nH]2)[nH]c(=NC2CCS(=O)(=O)CC2)[nH]1 c1(C(N2CC3CC(CNC(C45CC(CO4)C5)=O)C3C2)=O)c(F)ccc(F)c1F N1(C(C(C2CCOCC2)NC(C(C)CCN(C)C)=O)=O)CCCC2(CC1)CC2 C12CN(C(=NCCCCl)NCCS1)CCS2.c1(CC)cc(Cl)ccc1Cl c1(C(N2CCCC(C(C)O)C2)C(=O)NCC)cc(OC)nc(OC)c1.C1CO1 CP(C)(=O)c1cnn(CC(=O)NC2CN(C(=O)C3CC3)CC2N=[N+]=[N-])c1 c1(C(=O)NCC2CN(C(CCc3cnc(C)o3)=O)C(C)C2)cccc2ccoc12 c1(CC(=O)N(C(CC)COC)C)ccnc(O)c1 C(CC(C(C)(C)C)NC(c1cc2n(n1)CCC2)=O)N(C)C(C1CCC2(CC2)C1)=O C(=O)(C(C)(O)CC=C)NCC(CNC(C1C(C=C)C1)=O)CO C1(CNC(COCC(=O)NC)=O)CCC12CCN(C(=O)C=CC(F)(F)F)CC2 N1(C(C2C3(CN(Cc4c(Cl)ccc(C)c4)C3)C2)=O)CC(F)(F)C(F)(F)C1 C(=O)(C1=NOC2(CCOC2)C1)NCC1N(c2ncn(C)c(=O)c2)CC(O)C1 N1(C(c2c(CC)scn2)=O)CC2CC(C1)N2C(C1CCCSC1C)=O c1(C(=O)NC23C(CN(C(c4nn[nH]c4Cl)=O)C2)C3)cccc(Cl)c1[N+](=O)[O-] C(CCF)(C(=O)OC)NC(C1(CNC(=O)C=CC(C)CC)CC(=C)C1)=O Cc1cc(=NCc2ncsc2C)[nH]c(=NCc2cnc(Br)cc2C)[nH]1 C#CC1CCN1C(C1CCC1NC(c1cscc1CC)=O)=O c1(N2CC3C(C(N4CC(C)(CO)C(O)CC4)=O)C3C2)ccc2ncoc2c1 C1(C(=O)NC2CC3C(NC(CN4C(C)CCC4)=O)C3C2)OCCCC1(C)C N1(C(C(CCC)C(C)C)=O)CCC2(CCCN2C(c2cn(C)nc2OC)=O)CC1 N1(C(c2nc(COC)oc2)=O)CC2CN(C(=O)CCCC(C)C)CC2C1 CCC(C)C(C(=O)NCC(CCNC(C1(CCOC)CC1)=O)OC)OC C#CCCCCC(=O)N(C)Cc1ccccc1CNC(=O)C(CC)C(=O)OC C1(c2nc(C(C)NC)nn2-c2ccc(OC)nc2)CCC2CC1C2(C)C N1(CC(C(=O)C(N(C2CC(CC(F)F)C2)C)=O)(C)O)Cc2ccccc2C1 c1(C(=O)NC(C)CC2CN(C(c3cncc(N)n3)=O)C2)noc2c1CCCCC2 N1(C(C(CC)=CC)=O)CC(CNC(=O)CSCc2ccccc2)CC(C)(C)C1 CCC1=C(C(=O)NCC(O)CNC(c2cc(Cl)ccc2F)=O)SCCO1 N1(C(C(C)O)=O)CCn2ncc(S(C)(=O)=NC(=O)C(C)CS(C)(=O)=O)c2C1 C1(C(N2C(C)(C(=O)OC)CCC2)=O)CCN(C(=O)CN2CCCC2)C(C)(C)C1 CC1(C(N2CC(O)(CNC(=O)C3=C(Cl)CCC3)C2)=O)CC(C2CC2)=NO1 c1(C(=O)NC2C(C(C)C)N(C(C3CCC3(C)C)=O)CC2)ccc2nccn2n1 c1(Cn2c(NC(CCC(F)(F)F)OCC3CC3)nnn2)cc(F)cc2nc(S)[nH]c12 CC(C(=O)NOCC(N1CCCC(CF)C1)=O)N(C)C CCCC(C)(CCC)C(=O)N1CCCOC(CNC(C2OCCC2C)=O)C1 C(CC(C(=O)N(C)C)N1CCC(C(=O)NCc2cccs2)CC1)SC c1(CN2CCC(C(C)Cc3cccc(O)c3)CC2)ccc2c(c1)CCC2 N1(C(C2CC(C)OCC2)=O)CC2(C1)CN(C(c1cnn(C(F)F)c1)=O)C2 O=C1CC(CC(=O)NC2CCCCN(C(C34CCC(CC3=O)C4)=O)C2)CCCN1 C(=O)(C(C)(F)C(C)(C)F)N(CCNC(c1cc(C)sn1)=O)C C#Cc1cn(C)nc1C(=O)NC(C(=O)NOCC1CC2C=CC1C2)c1cccs1 c1(C(N2C(C)(CNC(=O)C(O)C(F)(F)F)CCC2)=O)cnn2c1OCCC2 C(CN=c1cc(NCCN2CCC(C)CC2)nc(-c2ccncc2)[nH]1)SCC c1(C(=O)NC(C)(C)CNC(c2ccc(Cl)o2)=O)ccc2c(C#N)c[nH]c2c1 c1(C(C)(C)C)cc2c(N(C3CNCC3O)Cc3ccc(CO)s3)ncnc2s1 c1(OC)c[nH]c(C(=O)NCC2CN(C(=O)C(C)N(C)C(C)=O)CC2C)cc1=O C=C1CC2(C1)CC(C(=O)NCC(C)NC(=O)CC1SC(=N)NC1=O)C2 Cc1cc(N)c(C(=O)NC2CCCN(C(=O)CCC(F)(F)F)C2C)nc1C c1(OCC)cc(N(C)CC2CCN(C(=O)C(C)NC(N)=O)CC2)nc(C)n1 c1(C(=O)NC2CCCN(C(C3CC(CCC)C3)=O)C2C)sc2nnc(S)n2c1C c1(CC(=O)NC2CC(CNC(C3CC3(F)Cl)=O)C2)ccc(O)cc1 c1(OC)ncc(-c2cnoc2C)cc1-c1ccnnc1 C1(SC)CCCCC1N=c1[nH]c2c(c(=NCCc3ncc(F)cc3F)[nH]1)COC2 N1(C(C(C)NC(N)=O)=O)CCCC2(CNC(=O)C(C)NS(C)(=O)=O)CCCC12 C#Cc1ccc(C(=O)NCC(C(=O)NCC(C)(COC)CC)C(C)C)cn1 CC1C(NC(=O)CN(C)CCO)CCN1C(c1nc(=N)cc[nH]1)=O c1(C(N2CCS(=O)CC2)C(=O)NCCSC)ccc(F)cc1F CC(C)(C)CCC(=O)N1CCC(F)CC1C(N1CCCC12CC2)=O C1(NC(C(CC)OC)=O)CCC2(CC1)CC(NC(=O)CCn1cnnn1)C2 n1(C(C)CO)cc(CN(C(=O)C(=O)NCC2CC(F)C2)C)nn1 C12(NC(Cc3c(Cl)cn(C)n3)=O)CCN(C(=O)CC3(C)CCC3)CC1C2 c1(CN(C)C(=O)NCC2CC3CCCCCCC23)nnc2n1CCNC2=O C1(C)(CCC)CCN1C(=O)CCCC1CCC1.C12CCN(C1)N2CC N(C1COc2c(F)cccc21)C(=O)NCCCCOC(C)C c1(C(C(=O)NCCCN(CCCNC(C2(C(F)F)CC2)=O)C)C)ccc(F)cc1 C(=O)(CC(C)C(F)(F)F)Nc1nc(C)c(SCC(N2CCCC(C#N)C2)=O)o1 C=CCCC(C(=O)NC(c1cnn[nH]1)C)NC(C1(F)CC1)=O N1(C(c2c(OC)ncc(Cl)c2)=O)CC2(CCN(CC(C3CCCCC3)OC)C2)C1 c1(C(=O)NC2(CCCC(=O)NCC3ON=C(C)C3)CCC2)ccc(C#N)c(C)c1 C(C)(C1CN(C(=O)OC)C=C1)=CC(c1n(CC)nnn1)NCCN(C)C(C)=O c1(C(N(CCCN(C(=O)C(F)CC2CCCC2)C)C)=O)cc(N)c(O)c(F)c1 c1(NCCC(C)(C)CO)ncc(S(=O)(=O)NCC2(CC)CCCC2)cc1Cl CC1CCC(CC(=O)NC(CC2CCC2)C(=O)NC2CC(n3cncn3)C2)CC1 N1(C(c2c(C)con2)=O)CCCC(NC(=O)C(F)(F)c2ccccn2)CC1 C(C(C)C(F)C(=O)NCc1nccn1CC)NC(CC)=O CC(CC1CC1)CN=c1c([N+](=O)[O-])c[nH]c2ccc(F)cc12 c1(CC#N)ccc(C(=O)NCC2CC(CNC(=O)Cc3cncnc3)CO2)cc1 C(CCCC(=O)NCC1CN(C(c2nccn2C)=O)CCO1)OC C1(C(=O)NCC2CC(C(=O)NCC3CC(O)C3)C2)CCCS1 c1(OC)ccc([N+](=O)[O-])c(CNC(=O)NCCC2(C)CCCO2)c1F c1(C(N(CC(=O)NCC2(C(=O)OCC)CC2)CC#C)=O)ccc(Cl)nc1 c1(CN2CCC(N(C(CCC3CC(OC)(OC)C3)=O)C)C2)cccc([N+](=O)[O-])c1 C1(N(C(C(F)=CCC)=O)C)CCCC2CN(C(c3ccc(Cl)cc3)=O)CC12 c1(CN2C(=O)C(F)NC(=O)CSCC2)ccc(Cl)cc1.C1(CC)CCCC1 n1(CCC)nc(C)c(C(=O)N(C)CC2C3CN(C(=O)C4=COCCO4)CC23)c1C C(=O)(C(CSC)C(C)(C)C)N(C1(CN)CCC1)C.C1(C(=O)OC)CN(C2CC2)C1 c1(C(N2C(C(N)=O)CCC2)=O)[nH]nc2ncc(-c3ccc(C(=O)O)nc3)cc12 C(=O)(C(O)C(C)(C)CO)OCCC1CCN(C)CC1 C1(F)(CNC(C(c2cccs2)SC)=O)COCCN(C(=O)Cn2ccc(C)n2)C1 CC(C)CCC(=O)C(=O)NC(C)(C)CC(F)C(=O)N1CCC(C)C1 N1(C(C(N2CC(C)C2)C)=O)CCCC1C(C)NC(c1csc(CS(C)(=O)=O)n1)=O Cc1nc(C(C)C)sc1C(=O)NCc1ccccc1CNC(C1(C2CC2)CC1)=O Cc1c(Cl)ccc(C(N2CCCC2C(C)(C)NC(c2ncn(C)n2)=O)=O)c1N Cc1ccc(SCC(=O)NC2CCOCC2NC(c2coc(C3CC3)n2)=O)cc1 Cc1cccc(-c2ccc(C(N3CC(CO)(NC(C4CCCOC4)=O)C3)=O)n2C)c1 c1(C(N2CC(CC)N(C(c3ccc(SC)o3)=O)CC2)=O)cnn(C)c1S(N)(=O)=O C(=O)(CC(C)(C)N(C(=O)COCC1CC1)C)N1CC(CCC=C)C1 c1(C(=O)NCC2COC(C(=O)NCC34CCC(C3)C4)C2)oc2ccccc2c1Cl c1(C(N2CCCC(NC(COCC(=O)OC)=O)C2C)=O)ccc2n[nH]c(C)c2c1Cl N1(N2CCNCC2)CCC(F)(CO)CC1.N1(C(=O)OCC)CCC(C=O)CC1 CCCCC(CC)C(=O)NC.C(=O)(CSC1CC1NC(C)C)NCC1(C(=O)OC)CC1 C(CCNC(c1nocc1C)=O)(C(C)C)NC(c1c(OC)scc1)=O N1(C(c2cc(C)c(Cl)cc2)=O)CC(C(N2CCC(O)C2C)=O)C(C)(C)C(F)C1 N1(C(c2cncc(OC)n2)=O)CC(O)CCC1C(=O)NC1(C)CCCC1C C1(N(C(=O)OC(C)(C)C)CCF)CCS(=O)(=O)C1.C12CCC(C1)C(=O)N2 C(C(=O)N1CCCC(OC)C1)(C(C)(C)C)NC(C(COC(C)=O)C)=O n1(CC=O)ccc(=NC(c2cc(Br)cc([N+](=O)[O-])c2O)C2CC2)nc1O C1(NC(C(c2scc(C)n2)C)=O)CC2CN(C(=O)CC(C)C3CCCO3)CC12 CC1CC(NC(=O)Cn2nnn(-c3cccs3)c2=O)CN1C(c1coc(Cl)c1)=O CC(C(C)C(=O)NC1(CCNC(C2(C(=O)C3CC3)CC2)=O)CC1)S(C)(=O)=O C(=O)(C#CC(C)(C)O)N1CCC(CC(=O)NCC#CCOC)CC1 N(C(=NCCOCC1CCCS1)NCC1CCCCO1)Cc1nc(C)on1 C1(C(=O)NC2(C)CC(NC(Cn3ncc(C)c3)=O)C2)OC2CCC1C2 c1(C=O)ccc(I)cc1NC.c12cnc(nc1)[nH]c2=O.C(=O)(NC)NCCNC(C)=O c1(C(=O)NCCCC(C)NC(CCNC(=O)NC)=O)cc(Br)c(C)s1 C1(CNC(CN(C(C)C)C)=O)(CNC(=O)CSCCC(F)(F)F)CCCC1 c1(C2CCN(C(C(=O)NC(CC)(C)C)C3CC3)C2)ccccc1F c1(C(=O)NC2CC(OCC(=O)NCC(CC)(C)O)C2)cnnc(C)c1 CC(CC(=O)N1CCC(C)C1CNC(c1ccc(Cl)c(Cl)c1)=O)CC(C)(C)C N1(C(C2CC(c3ccc(Br)cn3)C2)=O)CC2CC(CF)(CO2)C1 c1(C(N2C(CN(C(=O)CN(C)C(N)=O)CC)CCC2)=O)cccc2c1nnn2C N1(C(Cc2c(C)nccc2)=O)CCOC2(CCN(C(=O)CCCCC(N)=O)C2)C1 c1(C(=O)NC2COCCN(C(=O)C=C3CCOCC3)C2)ccc2c(c1)NCCC2 C(C(C(=O)NCC(C)N(C)C)C(C)C)NC(C1CC(OCC)C1)=O c1(OCC(=O)NCCN(C(=O)C=C2CCCC2)CCOC)cnn(C)c1 C1(OCC)CC2(C1)CC2NC(C1CC1CNC(C1(O)CC1)=O)=O C(=O)(C(O)C1=CCCCC1)N1CCN(C(C23C(C)(C)OCC2C3)=O)CC(CO)C1 Cc1c[nH]nc1CNC(=O)COC1CN(C(C2CCCC2C)=O)C1 C1(N)CCOC2(CCCC2)C1.c1(COCC(=O)NCC2(CO)CCC2)ccccc1 c1(C(N2C(C)CC(CC(F)(F)F)C2C)=O)cc(F)c2ccccc2c1 c1(C(=O)NC2C(CNC(C(C)=NOCC#N)=O)C2)ccc2cnn(C)c2c1 C1(CC(=O)N(CC(F)F)CCOCC(=O)NCCOC)CC12CC2 C1(NC(C)=O)CN(C(=O)CCc2c(F)cccc2Cl)C2CCCCC12 Cn1ncc(C2CC2)c1C(N1CC(CNC(C2COCCO2)=O)C(O)C1)=O CCC(C(C)C)NC(=O)CC(C)NC(=O)C(F)=C(C)C C(O)(CC(=O)N1CCOC2C(O)CC12)(C(F)(F)F)c1c(C)nccc1 N1(C(Cc2n(C)nnc2)=O)CCN(C(=O)C=Cc2nccs2)C(CC(F)F)C1 C1(NC(C=C(C)C)=O)CC2(C1)CC2Nc1ncc(I)cn1 c1(C(=O)NCC(C)CNC(=O)C(C)n2ccnn2)cccc(C(C)(C)C)c1 Cc1ccc(Cl)cc1C(=O)NCCc1cn(-c2cncc(Cl)c2)nn1 C(=O)(C(C)(C)c1csc(-c2ccccc2)n1)NCC(C)NC(=O)CNC=O CCC(CC(=O)NC1CC(CO)N(C(C2CC(CF)C2)=O)C1)C1CC1 C1(NC(c2ncc(OC)nc2)=O)CC2CC1CN2C(C1CSC1)=O N1(C(Cc2cnc(C)s2)=O)CCCC(NC(C2CC3(F)CC2C3)=O)C1 CC1CN(C(C2CC2C2CCC2)=O)CCN1C(=O)COc1ccc(F)cn1 C(=O)(CCCC(C)(C)C)OCCN(C(CC)C)C CC(C(C)C(=O)NCC1C=CCOC1)NC(=O)CN(C1CCC1)C c1(NC(c2n(CCC)nnn2)(C)CCCl)ccc(Cl)c(CC2CCCCO2)c1 N1(C(C2CCC(CNC(=O)CCC3CCCCC3)C2)=O)CC2CC3CC2C1C3 C12(CCOCC1)N(C(=O)CC1CCC1)C2.C(=O)(C(F)=CCF)NCC(F)F C1(NC(=O)C2=CCCO2)CC1C1CCCN(c2ncnc3[nH]ccc23)C1 c1(C(=O)NC(CCNC(C(c2ccccc2)OCC)=O)C)cc(C)sc1Br C(N=c1[nH]c(=NCc2nncs2)[nH]c2c1CCC2)c1[nH]c2ccccc2n1 C(CCC(O)C(=O)NCc1ccccc1F)NC(c1c(C)noc1)=O Cc1c(C(=O)NC2CCN(C(=O)CNC(N)=O)CC(C)(C)C2)nn2c1CCCC2 S(=O)(=O)(c1ccc(Cl)cc1Br)NC1C(C)OC2(C1)CCC2 C1(C(N(CCCC)CCCC)=O)CN(C(=O)C(C)CCC)CCC1(C)C N1(C(C2CCC(F)(F)CC2)=O)CCC(C2(N=c3ccn4nccc4[nH]3)CC2)CC1 c1(C(N(CCCN(C(=O)CSc2ccc(O)cc2)C)C)=O)cnc2sccn12 N1(C(C(CC)SC)=O)CC23CCCC2(C1)CN(C(c1cnc(F)c(C)c1)=O)C3 C(=O)(CCC1=CCCCC1)NC1C(NC(c2n(C(CC)C)ncc2)=O)COCC1 N1(C(c2c(C)nn(C(C)C)c2)=O)CCCC(CO)(NC(=O)CCC(C)N(C)C)C1 c1(OC)cc(C(c2nnnn2C2CC2)NCC2(CF)CCC2)c(F)cc1F.C(C)(C)O C12(CNC(c3c(CC)cccc3F)=O)CN(C(c3cn[nH]c3)=O)CC1CCO2 Cn1cc(C(=O)NC2CC3CN(C(=O)C4=CSCS4)CC23)n(C)c1=O C(C)(C)(CC(=O)NCc1cn(CC(=O)NC2(F)CCOCC2)nn1)OC Cc1ccc(Cl)c2c1CCCN2C(=O)N(C)C(C)C1CC1 C(=O)(C(C(C)CC)N(C)C)NCC(C)N(C(c1cnn(CCO)c1C)=O)CC C1(C(=O)NC(CNC(C(=O)NCCO)C(C)C)(C)C)(CC)CC(C)(C)C1 Cc1csc(C(=O)NC2CC(n3cc(CCC(C4CC4)N(C)C)nn3)C2)c1 c1(C(=O)NC2(CC(=O)NCCOCCC=C)CCC2)cc(O)c2ccccc2c1 CCC(O)(CN(C)C(c1cn(CCNC(c2ncnn2C)=O)nn1)=O)CC C#Cc1ccc(C(=O)NC2(C(N3CC(N4CC(=O)NC4=O)C3)=O)CCSC2)o1 C(=O)(C(C)(F)C(=O)NC1CC(NC(=O)C(C2CC2)SC)C1)OCC c1(C(=O)NC23CC(NC(CC(=O)OCC)=O)C(OC2)C3)cc2n(n1)CCCC2O c1(C(=O)NCC(CC)NC(=O)CC2CC(O)C2(C)C)cnc(C2CCC2)cc1C C1(C(=O)NCC2CC(NC(C3C(CC)OCCC3)=O)C2)CCCC2(CCC2)O1 CCC(C(=O)OC)C(=O)N1CCCC1(C)C(N1CCC(C(C)OC)CC1)=O N1(C(CCNC(N)=O)=O)CCC(NC(c2ccc(F)cc2)=O)C(CO)CC1 C=CCC(CC(=O)N1CC=CC(O)C1)NC(c1cc(C)oc1CC)=O C(=O)(CC1CCCc2ccccc21)N1CC(CNC(C2(CC)CC2)=O)S(=O)(=O)CC1 C1(N(C)C)CCn2cc(C(=O)N(C)C(c3cn(CCCC)nn3)C3CC3)nc2C1 C1(NC(=O)CCN2CCC(F)C2)CCN(C(=O)CCC2CC2)C12CC2 CC(C(=O)N(C1(CNC(C2(CC3CC3)CC2)=O)CC1)C)=C1CCCC1 C1(C(=O)NCC(CN(C(=O)Cc2ccsc2)C)(C)C)Cc2cc(F)ccc2O1 c1(C(N2CCC3CN(C(C4(c5cccs5)CC4)=O)CC23)=O)ccc2c(c1)C=CCC2 N1(C(c2cccc(=S)n2O)=O)CCC(NC(C2(F)CCOC2)=O)C2(CCC2)C1 c1(C(=O)NCC2(F)CC(NC(C3CC(OC)C3)=O)C2)cccc2cc(Cl)ccc12 c1(CC)cc(C)ccc1C(=O)NCC=C1CCN(C(=O)CC(C)(O)C2CC2)CC1 N1(C(C(=O)NCCOC)=O)CCC2(CC1)CC(C)N(C(C1C3CCN1CC3)=O)C2 C(=O)(C1=NOC2(CCOC2)C1)NCC1(C)CCN(C(c2scc(Cl)c2Cl)=O)C1 CCS(=O)(=O)CCN1CCN(CCn2ccc(C(F)(F)F)n2)CC1 CC(N=c1[nH]ccc(C#N)c1Br)c1cnc(C(C)(C)C)s1 C1(C(NC(=NCc2ccc(F)cc2)NC2CCCC(F)C2)C)CCC(F)(F)CC1 c1(SC)cccnc1C(=O)NCC1CCCC(CNC(=O)C(C)SC(C)C)C1 Cc1cnc(CCNC(c2sccc2CNC(C2(C)CCCOC2)=O)=O)nc1 c1(NC(C2CC3(C2)CN(C(c2ccnc(Cl)c2Cl)=O)C3)=O)cnc(Cl)c(CO)c1 CCCC(C)(CC)C(=O)N(CCN(c1ncno1)C)C(C)C N1(CC)CC(C(=O)N2CCC(N(C(=O)CCC(C)(F)F)C)C2)c2ccccc21 CC(CC(N)=O)C(=O)NCc1nc(CNC(c2c(O)cncc2F)=O)cs1 Nc1cccc(CC(N)C(=O)NCN)c1.C12CCCC1C(=O)N2 C1(SC)CN(C(c2cc(Cl)cnn2)=O)CC1NC(=O)C(C)(C)n1cnnn1 C1(NC(COCCCOC)=O)CCOCC1NC(=O)CS(N)(=O)=O O=S(=O)(c1ccc(CC(F)(F)F)cc1)NCC(O)C(F)F c1(C(=O)NC(CCNC(Cn2nnc(C)n2)=O)C)cccc2ccnn12 CC#CCC(C(=O)N1CC(C)(F)C1)NC(=O)CN1CCOC1=O CCC(C(=O)NC12CC(C(=O)NCC3CCCC4(CC4)C3)(C1)C2)C(C)(C)CC n1(CC(=O)NCC2(C(C)NC(C(CO)OC)=O)CC2)c(C)ccc1C CN1CCN(C(c2cnc(S)n2C)=O)C(CNC(c2nccnc2N)=O)C1 c1(C(=O)NCC2CC(NC(c3n(C=C)nnc3)=O)C2)cc(C)cc(C)c1N C1(CC(=O)NCC(CC2CC2)C(=O)N2CC(n3cnnc3)C2)CC2(CCC2)C1 Cc1cc(NC(C2CC3CCC3N2C(=O)CCC2CCCOC2)=O)cc(C)c1C Cc1ncc(C(=O)N(C2CCN(CCO)CC2)C(=O)C#CC(=O)O)cn1 c1(OC)cccc(C(=O)N(C2CN(C(=O)CCSC(F)(F)F)CC2F)C)n1 c1(CN2CC(C)N(C(c3cc(Br)ccc3C#N)=O)CC2)cnc2ccc(F)cn12 CC1OC2(CO)CC1(C(=O)N(CCC(C)NC(c1cccnc1O)=O)C)C2 N1(C(CNc2cn(C)nc2)=O)CC(NC(C2COCCO2)=O)CC2(CC2)C1 C1(NC(C(CC)(C)C)=O)CC2CC(C1)N(C(c1csc(C(C)(C)C)n1)=O)C2 c1(C2(C(C)C)CC(C(=O)NCC(=O)N(CC(C)OCC)CC)C2)ccc(F)cc1 c1(CC)cc(=NC(=O)C23CC4CC2C3C4O)[nH]n1C.N12CCN(CC1)C2=O c1(C(=O)NC2CCCCN(C(C3C(OC)CC3)=O)CC2)cccc(Cl)c1[N+](=O)[O-] C(=O)(C(=O)C(C)CC)N1C(CC(=O)NC(CCCC)COC)COCC1 CC(C)C(O)CC(=O)N1CCC(CO)C(NC(C2CC2c2cccnc2)=O)C1 C1(CNC(C2CCCS2)=O)CCN(C(C2CC2F)=O)C1 N1(C(CC(C)(F)F)=O)CCN(CCC2(NC(N3CCCC3)=O)CC2)C2(CCC2)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1(F)COc2ccccc2O1)NCC(OC)OC Cc1nccc(C(=O)NCC2CN(C(c3cc(Br)nn3C)=O)CCO2)c1N N1(C(c2c(CC)noc2C)=O)CCC(C)C(N(C)C(c2cccc(Cl)c2F)=O)C1 CC1(F)CN(C(=O)Cc2ccns2)CCN(C(C2CCC(N=[N+]=[N-])C2)=O)C1 CCCC(C(=O)N1CCOC(C)(CNC(c2cncn2C2CC2)=O)C1)S(N)(=O)=O c1(C(=O)NC2CN(C(CCC(=C)Cl)=O)CC2O)cc2cccc(C)c2s1 c1(C(N2CC(CN(C(=O)CCSC3CCC3)C)OCC2)=O)ccn2ccnc2n1 Cc1ccc(C)c(CNC(=O)NC2(CC3CCC3)CCC2)c1 Cc1cc(C(=O)N(C(C)CNC(C2(C)CCNC(=O)C2)=O)C)cc(C)n1 c1(C(=O)OCC)[nH]c(=NCCN(C)C(c2cc(Cl)cn2CC)=O)sc1C Cc1ocnc1CC(=O)NCCCN(C)C(C1CCC(c2cc[nH]n2)O1)=O C1(O)(CCNC(=O)C2=C(Cl)CC2)CCCN(C(c2cc[nH]c2C2CCC2)=O)C1 C1(NC(c2nccc(C)n2)=O)CCC2CC1CN2C(=O)C=CCF CC1Cn2nccc2CN1C(=O)CCN(CCO)C(c1cccc(F)c1O)=O c1(CC(N2C3C(CNC(C4CCS(=O)(=O)C4)=O)C(C3)C2)=O)cc(F)c(F)cc1F C1(O)(CCNC(CCOC(C)C)=O)CCN(C(=O)C(C2CCCCC2)C)C1 S(=O)(=O)(c1ccc(N(C)CCO)c(F)c1)Nc1ccc(CNC2(SC)CC2)cc1F N1(C(c2sccc2Cl)C(=O)NCCCF)CCCCC(N2CCCC2)C1 CCC(C)C(C)C(=O)N(CCCCN(C(=O)Cc1csc(-c2cccs2)n1)C)C C(CCCCCC(=O)N1CCC(N(C)C(c2csc(C(C)=O)n2)=O)C(C)C1)SC C#CCC(C)(C)C(=O)NCC12CC1CN(C(c1c(C)nn(C)c1Br)=O)C2 C1(CNC(C(=O)NCC)=O)CN(C(c2ccc(N)cc2O)=O)CC12CCC2 c1(C(N2C(CCNC(CCOCC(C)C)=O)CSCC2)=O)ccn2cccc2c1 C(C(CO)N=c1[nH]nc(C(C)C)o1)NC(c1cc(CC)n(-c2ccccc2)n1)=O C1(NC(c2ccc(CO)o2)=O)CCC12CN(C(=O)CCC1CCOCC1)C2 N1(S(C)(=O)=O)CCC(CNC(=O)CCC(=O)N2CCCC(N(C)C)C2)CC1 Cc1cc(CNC(=O)NCC2CCS(=O)(=O)N2C)nc(Cl)c1Br c1(CNC2CN(C(c3cc(C)nn3C(F)F)=O)CC2O)cc(F)cc(Br)c1 C#CC1CN(C(c2cc(O)ccc2C)=O)CCN1C(C12CCCC1C2(F)F)=O C1(C(N(CC(CN(C(=O)CCCCc2cnn[nH]2)C)O)C)=O)CCCCC1(C)C c1(C(C)=O)cc(Br)c(C)cn1.C12CN(CCS1)C(=O)NC2 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(CCNC(C2CCCC23CC3)=O)CCC1 c1(C(=O)NCCN(C(CC(=C=C)C)=O)C)ccc(-c2ccncc2)cc1C C(=O)(C(C(F)(F)F)C(F)(F)F)N(C1CCN(C(C(CCCC)C)=O)C1)CCO N1(C(c2cnc(SC)nc2O)=O)CCC2C(C1)CN2C(=O)C1=CC(C)(C)C1 N1(C(C(CCOC)NC(=O)C(CO)OC)=O)CCCNC(=O)C1C N#Cc1ccnnc1NCC1CC2(CC(NC(c3coc(O)n3)=O)C2)C1 Cc1c(F)cc(C(=O)NCC(CNC(c2cc[nH]n2)=O)CO)c(F)c1N C12(NC(CCc3c(C)noc3Cl)=O)CCCN(C(=O)C(C)(C)O)CC1C2 Cc1nc(CCC(=O)NC2CC(CNC(=O)Cn3nnc(=N)[nH]3)C2)oc1C N1(C(C2N(C)CCC2)=O)CCCN(C(=O)Cc2ccc(C(F)F)cc2)CC1CO C12(C(=O)NC(CCC(N3CC(COC)OCC3)=O)C)CCC(C1)OC2C N1(C(C(CC(C)C)ONC(c2cc(=NC)[nH]cc2)=O)=O)CCOC2CCCC12 N1(C(c2c(C(=O)OC)c(C)on2)=O)CCC(NC(c2cc(C)nn2C)=O)C(C)C1 N1(C(C2(CC)CCC2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(O)CC(C)(C)C N1(C(CCSC)=O)CCOC(CN(C(=O)Cn2c(O)nnc2O)C)C1 C1(C)(NC(c2cnc(C)o2)=O)CCN(C(c2cccc(CC#N)c2)=O)CC1 c1(CC)[nH]nc(C(=O)NCCCCC2CN(C(c3nnn(CC)c3C)=O)C2)c1Br C1(C#N)(C(=O)NCCCCC(N2CC=C(C)CC2)=O)CC2CC2C1 C(C(CC(C)C)C(=O)N1CCC(CC(=O)NC(C)CN(C)C)C1)OC c1(C(=O)NCC2(O)CCN(C(c3cnccn3)C)CC2)coc2c1C(=O)NCC2 N1(C(c2cccc(OC)c2)=O)CCCC2(NC(c3cc(O)nc(Cl)c3)=O)CC2C1 c1(C(C)NC(CN(C2CC2)CC)=O)ncnn1C.C1(C(=O)N(C)C)CC(CF)C1 N1(C(C2CCC(C)N(C(=O)Cn3[nH]cnc3=N)C2)=O)CC(C#N)C2(CCC2)C1 c1(CC)ccccc1CC(=O)NCC12CC1CN(C(c1ocnc1C)=O)C2 N1(C(c2cccc(C)c2N)=O)CC2CC(C)N(C(=O)CC3CCC(C)(C)C3)C2C1 N12CCC3CC3(CC1)C(=O)Nc1cc[nH]c1C2=O.c1(C2CN(CC)C2)ccncc1 C(=O)(C#CC(C)(C)O)NCC12C(CN(C(C(C)OC3CCOC3)=O)C1)C2 CC1CN(c2ccccc2CNC2CCCCC2NC(=O)C2CC2)CC(C)O1 c1(C(N2CCC(NC(c3ccc(O)cn3)=O)(CO)C2)=O)cc2ccc(Cl)cc2[nH]1 O=C1CCC(CC(N2CCC(CCn3cc(-c4cncnc4)nn3)CC2)=O)CN1 C(=O)(C(C(C)C)C(C)C)NCC1C2CN(C(Cc3cccc(C)c3)=O)C(C2)C1 C1(C(N2CC(CNC(CNC(CCC)=O)=O)C(O)C2)=O)CC(=O)NC(=O)N1 C(CCN(C)C(C1CCCCS1)=O)(C(C)C)NC(C1(OCC)CCOC1)=O Cc1cccc2[nH]c(C(N3CCCCC3CNC(c3cccc(O)n3)=O)=O)cc12 Cc1ccccc1C=CC(N1CC2(NC(c3cc(C)n(CO)n3)=O)CCC1C2)=O N1(C(CSCC)=O)CCC2(CNC(=O)C=Cc3ccccc3)CCCCC12 O=C(C#Cc1ccccc1)N1CC2CCCN(C(c3ccnc(Br)c3F)=O)C2C1 CC(CC(=O)NC(C)(C)C(C)NC(c1ccc(Cl)cc1)=O)C(F)(F)F c1(CC(=O)N(C(C)CN)C(=O)Cc2cnsc2)ccc(O)nc1.CO N1(C(c2cc(OCC)ncc2)=O)CC2CN(C(C3COCC(C)(C)O3)=O)CCC12 N1(C(C2CCC(CC(=O)OC)O2)=O)CCC(NC(c2ccc(F)cn2)=O)C(O)C1 c1(C(N2CCN(CCF)CC2)=O)ncc(-c2ccc(O)cc2C(F)(F)F)cc1F N1(C(=O)Cc2cncs2)CC2CCC1CN2C(=O)C=C1CCCCCC1(F)F CC1CC(NC(C2CCC2(F)F)=O)CN(C(c2cnc(C3CCC3)nc2O)=O)C1 c1(C(=O)NC2CN(C(c3cnn(C)c3N)=O)CC2(C)C)coc2c1C(=O)NCC2 CC1CCc2onc(C(=O)NCC#CCNC(c3ccnc(S)c3)=O)c2C1 N(C1CCOc2c(OC)cc(C)cc21)C(=O)NCC(C1CCOCC1)CC C(=O)(CC(C)(C)C)N1CC(C(C)NC(C2COC(=O)N2)=O)C1.C1(=O)CN1 c1(CC(=O)NCC(C)N(C(=O)CCNC(C)=O)CC)ccsc1Br C(C1=CCN(C(c2cc(C(F)(F)F)no2)=O)CC1)NC(Cn1c(C)csc1=O)=O N1(C(c2cc(CC)c(C)s2)=O)CCC2CN(C(c3ncc(Cl)cc3F)=O)CC12 C(C1=NOC2CN(C(C3C4COCC34)=O)CC12)NC(c1cc(C)c(C)[nH]1)=O C1(C(N(CC(O)CNC(=O)CCc2cnn(C)n2)C)=O)CCCC(N(C)C)C1 C1(NC(c2c(CC)cccn2)=O)CCN(C(C23CCOC(C)(C2)C3)=O)CC1C S(=O)(=O)(c1ccc(I)cc1)N1CC(NC(C(CCCCC)C)=O)C2(C1)CNC2 C1(CN(C(=O)Cc2ccc(Br)cc2)C)CN(C(=O)C(F)C(C)(C)O)CC12CC2 C=CCCC(C(=O)NCC1CCOC1C)NC(c1nnsc1C)=O c1(C(=O)NC2CCCN(C(Cn3ccc(C)n3)=O)CC2)c[nH]c(=O)c2ccnn12 Cc1cc(=NC2CCN(C3CCOC3)CC2)[nH]c(=NCCCOCCN(C)C)[nH]1 C1(O)(C(C)NC(=O)COC(F)F)CCN(C(c2cnn(C3CC3)c2)=O)C1 CC(CC(F)F)C(=O)N1CCN(CC(C)(C)NC(=O)CSc2ccncc2)CC1 CC1(C)CC(CNC(C23CC(CSC4CCOC4=O)(C2)C3)=O)c2ccccc2O1 C(c1cccc(C#N)c1)=CC(N1CCCC(NC(C2(C(N)=O)CCC2)=O)CC1)=O N1(Cc2c(C)nc(C)o2)CCC(C)C(NC(c2snnc2C(C)C)=O)C1 c1(CNC(N2CCOCC2)C(=O)NC(C(=O)OC)C)[nH]nc2ncccc12 Cc1cncc(C)c1C(N1CCOCC(CNC(=O)COc2cnn(C)c2)C1)=O c1(C(C)(C)C)n[nH]cc1C(c1nnnn1Cc1cccs1)NC1CC(CO)C1 CC(C(=O)OC(N1CC2CC=C1C2)=O)(C(F)(F)F)c1ccccc1 CC(O)C(C)C(=O)N(CCCOCCNC(c1ccccc1F)=O)C.CCC CC(C)(C)C(O)C(=O)N1CC(NC(C2CCCC(=O)C2)=O)C(C)(C)C1 c1(C(c2nnnn2CCCOCC)NC(C=C)C2CC2)cc(C)c(F)cc1Br c1(C(=O)NCCCNC(c2cnc(OC)s2)=O)ccc2c(c1)CC(C)O2 CCCCS(=O)(=O)CC(=O)NC1CC(NC(C2CC(O)(C(F)F)C2)=O)C12CCC2 C(=O)(C(C)CC(=O)NC(CNC(=O)CC1=CCCC1)CC(C)C)OC N1(C(c2cnc(CC)s2)=O)CCN(C(c2ccon2)=O)C(CCO)C1 N1(CCC)CCC(F)(F)C1.N12CC(C1)NC(=O)C(=O)N(C)CC2 N1(C(C(C)O)=O)CCC(NC(c2cc(Cl)ns2)=O)C1C(C)C C1(NC(c2cc(COC)on2)=O)CC(O)CN(C(=O)CCc2cccc(Cl)c2)C1 C1(C(=O)NC2CCC(C(C3CCCC3)NC(c3c(C)scn3)=O)C2)C(C)(C)C1(C)C CC(C(=O)NCCC1(CN(C(=O)C(F)n2ccnc2)C2CC2)CC1)NC=O.CC c1(C(N(CC(C)C(=O)NCC(c2ccco2)O)C)=O)c[nH]c2ncccc12 Cc1ccc(C(C)C(N2CCCC2C2CCCOC2)=O)o1 CCC(C)C(O)C(=O)N1CCN(C(c2cc(CC)cc(F)c2)=O)CC1C1CCC1 C#Cc1cnn(C)c1C(=O)NC1CCCN(CC(F)(F)F)C1=O NC(Cc1ccccc1)C(=O)NC(C1CCC1)C1CC1 C=CC1(O)CCN(C(=O)C(N)CC2CCOC2)C1 CC(C)(C)C(CNC(c1cc(O)cn1C)=O)C(=O)N1CCCC1(C)CCCO C(CCS(C)(=O)=O)N(C(CCN(CC#C)C(c1cnn(C)c1OC)=O)=O)CC C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C2CC(NC(C3CC(=C)C3)=O)CC1CC2 N1(c2ccc(NC(=O)NC3(c4cccc(C)c4)CCOCC3)s2)CCS(=O)(=O)CC1 C1(NCCSC(C2CCCC2)CC)CCOCC1 n12nnnc1C1(CCC1CS(C)(=O)=O)NCCC2.c1(CC2(C)COC2)ccccc1 CN1C(=O)OCC12CN(C(=O)C(F)(F)c1ccsc1Cl)C2 c1(CN(C)C(=O)OC(C)(C)C)ncc(C(=O)NCC23COC(C2)C3)cn1 S(=O)(=O)(c1cnc(NCC2(Cl)CC2(F)F)c(Cl)c1)NCC(C)N(C)C C1(CCC(=O)NC2(CC=C)CCOC2)CCCCN1C(=O)CC1CCCC(C)C1 c1(C(=O)NC(CCOC)CNC(=O)C=Cc2cnccn2)cc(F)cc(N)c1F c1(-n2cc(CC3N(C(C4N(C(C)=O)CSC4)=O)CCC3)nn2)c(Br)cnn1C Nc1cc(C(N2CCN(C(c3csc(Cl)c3)=O)C(CC3CC3)C2)=O)cc(F)c1 C(C)(C(=O)N(C(C)CN(C)C)CC)(C(C)C)NC(c1c[nH]c(=NC)s1)=O C12(C(=O)Nc3c(C)ccnc3Cl)CCCC1CN(C(=O)CSc1nc[nH]n1)C2 N1(C(C(C)CC2CC2)=O)CCCC(N(C)C(C2(Br)CC2)=O)C1 C(CC(C)C)(C(=O)NC)n1c(C(CC)(C2CC2)NCCC2CC(C)C2)nnn1 Cc1ccc(C(=O)NCC2C3CN(C(c4n[nH]cc4Cl)=O)CC23)c(=O)n1C Cc1cc(C(=O)NC23CC(NC(C4(C)CCCCC4)=O)(C2)C3)c(Cl)cc1F C=CCCN=C(NCC(N1CCOCC1)C)NCC(O)C1(C)CC1 c1(OC)cccc2c(C(N3CCCC(CNC(=O)CCC(C)(F)F)C3)=O)coc12 C1(CNC(C2CC(C)(CC)C2)=O)CN(C(c2c(C)cnn2C)=O)CC2(CCC2)O1 N#CC1CC2(CC(NC(C3CC(NC(=O)C(F)C(F)(F)F)C34CCC4)=O)C2)C1 c1(C(=O)NC2CN(C(CSC(C)C)=O)C3C2C3)cnc2cnn(C)c2c1 C#CCCC(C(=O)NCC1C=CCCC1)NC(=O)CCn1cc(C)cn1 CCC(CC)C(C(=O)NCCCC1CCCN1C(c1ccco1)=O)OC N1(C(COCc2cc(C)no2)=O)CCC(NC(=O)C2=CCCS2)C(CO)C1 c1(CS(Cc2scc(C(C)=O)n2)=O)cccc(C)c1C Cc1cccc2c1OC(C(N1CC3CCCCC3(NC(=O)C(N)=O)C1)=O)C2 N1(C(c2c(OC)cncc2)=O)CC2CCC1CN2C(C1CC2(C1)CC(C)C2)=O N1(C(c2c(CC)noc2C)=O)CCOC2(CCN(C(C3(O)CC3(C)C)=O)C2)C1 C(=O)(CCCC(C)(C)C#N)NCc1c(C(=O)NCc2c(C)cccc2C)nco1 c1(C(=O)NC2CCC(OC)C2)ccccc1Cl.c1(C(=O)N)sccc1CC#N N1(C(C=C(C)c2ccco2)=O)CC(F)(F)CC1CNC(=O)Cn1ccc(C)n1 c1(C(N2CCN(C(C(COC)C)=O)C(C)CC2)=O)cc(OC)cc2c1OCC2 C1(NC(c2cc(CC)oc2C)=O)CCCC(NC(=O)C(F)C2CCCC2)CC1 CCC(CC(=O)N(CCNC(C1CC(C(C)C)C1)=O)CC1CC1)c1ccccc1 c1(C(N2CCC(C(C)NC(C(CC)F)=O)C2)=O)cc(N)ccc1O CC(CC(=O)NCC1COC(CNC(=O)Cn2nc(O)ccc2=O)C1)P(C)(C)=O CC1(C)CCCOC1C(=O)NCCC1CCCN1C(c1cccs1)=O c1(CNC(C2CCN(C(=O)NC(C)C)C2)=O)cccc(CN=[N+]=[N-])c1 c1(N2CCN(C(c3ccccc3Cl)C(=O)OC)CC2)ccnc(C#N)c1 N1(C(C(COC)NC(C(CC)NC(C)=O)=O)=O)CC2CC=CCC2C1 N1(C(C)C)N=C(C(=O)N2CCOC(CN(C(=O)CCCC(F)F)CC)C2)CCC1=O CCC(C)C(O)C(=O)N1CCOC(CNC(=O)CSCc2csc(=N)[nH]2)C1 Cc1ccc(OCC(N2CCCC2(C)CNC(=O)CN2CCCC2C)=O)c(C)c1 C1(C(=O)NC(C2CCCC2)CNC(c2cncc(F)c2)=O)CC2(C1)CC2F C(=O)(C(CNC(C1CC(O)C(F)C1)=O)C(C)C)NC(c1cc(C)no1)(C)C C1(C(=O)NCC(CNC(c2cnc(CCC)s2)=O)CO)CC12CCOCC2 Cc1nc2sccn2c1C(=O)NCC#CCNC(C1CC2CCC1C2)=O c1(CNC(=O)Cc2ccc(F)c(Br)c2)ccc2c(c1)CNCC2 N1(C(C(N2CCOCC2)C)=O)CCC2(CCCC2NC(C2C(C)(C)C2(C)C)=O)CC1 N1(C(c2ccc(NS(CC)(=O)=O)cn2)=O)CCC2(CCCC2NC(=O)C(N)=O)C1 N1(S(CCCC)(=O)=O)CCC2(CC(C(=O)Nc3cc(C(=O)O)c(Cl)cc3F)=NO2)C1 C12CCc3ccccc3C1NC(=O)CCN1C=CC(=NC2=O)N1.CNC c1(OC)nc(C)ccc1C(=O)N(CC(C)(C)NC(=O)CC1CC2(CCC2)C1)C O(NC(=O)C(=O)N=c1cnn(CCc2ccccc2)[nH]1)C(C)(C)C Cc1cc(=NCCC23CCCN2CCC3)[nH]cc1S(=O)(=O)NCC12CC(CO1)C2 N1(C(C(CSC)O)=O)CCN(C)CC1C(N1CC([N+](=O)[O-])C1)=O CC1CCCC1NC(=O)NCCN(C)CC1CCOCC1 C1(C)(C(=O)NC(c2ncc(C)o2)C)CCN(C(c2nnn(C)c2C)=O)C1 C1(O)(NC=O)CCCN(C(N)=O)C1.Cc1ccncc1CNC1C(C(C)(F)F)C1 C1(NC(c2ccc(CCC)cc2)=O)CN(C(=O)C(O)CC)CC2(CCC2)C1 c1(CNC(=O)N(CCCOC)C)ccc(OCCOC)c2ccnn12 c1(C(C)(CC2CCOC2)NCC(=O)NC2CCC2)nnnn1CCn1cncn1 c1(C(=O)NCC(CC=C)NC(c2scc3c2OCCO3)=O)cc(Cl)cnc1C CN1CCC(c2ncc(C(=O)NCCCn3cc(C4CC4C(=O)O)nn3)[nH]2)CC1 C1(C(C)C)CN(C(c2nnn(C)n2)=O)CCCN1C(C1(C(F)(F)F)CCC1)=O c1(C(N2CCN(C(Cc3cccc(CC)c3)=O)CC2C)=O)cnc2c(c1)NCC2 N1(C(C)=O)CCC2CCN(C(C3(C)CC(F)C3)=O)CC2C1.c1ccncn1 C(CCC(N)=O)(C(=O)N1CC=CC(NC(c2cc3c(s2)CCOC3)=O)C1)N(C)C CCCCC(C(=O)N1CCC2(CC=CCO2)C1)C(C)C c1(C(=O)NCCC2(OC)CN(C(=O)CC(C)N(C)C)C2)c(C)cc(O)nc1C C(C(O)(CNC(C1CCC(NC(c2ccc(C)nc2)=O)C1)=O)CO)OC c1(C(N2CCC(C3CCCO3)C2)C(=O)NC2CCC2)cccc(Br)c1F C(CCNC(c1cn(C2CC2)cn1)=O)(C(C)C)NC(c1ncn(CC)n1)=O C1(CNC(=O)CC=C(Cl)Cl)CCCC2(CN(C(=O)C=CC3CCC3)C2)O1 C1(C(=O)NCC2(F)CN(C(=O)CNC(=O)C3CC3)C2)SC2C=CC1CC2 N1(C(N2CC(CCC)C(NC(c3cnc(OC)cn3)=O)C2)=O)C(=O)CN(C)C1=O N1(C(C2CCCO2)=O)CCC(N(C(C2CC(C(F)F)C2)=O)CC2CC2)CC1 Cc1nn2cc(C(=O)N(CC3=CCSC3)C)cnc2c1Br c1(C(=O)NCC(C)CNC(C2Cc3nccn3C2)=O)cc(F)cc2nc(S)[nH]c12 C1(CNC(C(C)OC2CCCC2)=O)(NC(c2ccc(O)c(Cl)n2)=O)CCCCCC1 C1(O)(CNC(C(C)(F)F)=O)CCCN(C(=O)CN2CCC(C(N)=O)CC2)C1 c1(C(=O)N(C2CCC(O)C2)CCOCCN(C)C(=O)C2CC2)cccc(C(F)(F)F)c1 c1(OC)cccc(C(=O)NC2CCCC2NC(=O)C(C)(C)n2cccn2)c1O.C(C)(=O)O c1(C(N2CCC(NC(C34OC(C)C(C3)C4)=O)C(F)C2)=O)noc2c1COCC2 c1(C(=O)NC(c2c(C)cccn2)C(C)C)cc(F)cc(F)c1N C(=O)(C(C(C)(C)C)OCCO)N(CC(C)O)CCNC(c1c(CC)n(C)nc1)=O N1(C(CCN(C)CCO)=O)CCC2(CC1)CC2(CO)CNC(=O)C1=CCCC1 C(=O)(C(C(C)(C)C)OC(C)(C)C)NCC(CCOC)NC(c1csnc1C)=O C1(C(C(=O)NCCN(C)C(C2CC2(C)C)=O)Cc2ccccc2)CCC(F)(F)CC1 Cc1sc2ccc(F)cc2c1C(=O)NC(CC(C)(C)C)c1ccc(Br)cc1 c1(C(=O)NCC2N(C(CC(C)C(F)F)=O)CC2)ncn2ccccc12 CC(C)CC(C)C(=O)NCC1CCCC1NC(=O)CC(C)(C)Cc1ccccc1 C(=O)(CCP(C)(C)=O)N1CCC(O)(C(C)NC(CSCC#C)=O)C1 C1(C(=O)NC2CC(NC(c3cccc(F)c3C(F)F)=O)C2)CCn2cncc2C1 c1(NC(C)C)ccc(C(N2CCC(CN(C)C(C34CC(C)C3C4)=O)C2)=O)cc1 C1(NC(N2C(C(C)(C)O)CCC2)=O)CCCCC(F)(F)C1 C(C(CC)(CC)C(=O)NCCCCC(=O)OCC)NC(CCC(CC)C)=O Cc1cc(CC(=O)N(C2CC(NC(c3ccc(F)c(F)c3)=O)C2)C)cc(C)c1 c1(C(=O)NCC2(F)CC(NC(c3cc(CC)ncn3)=O)C2)ccnc2cc[nH]c12 c1(C(N2CCN(C(CC=C)=O)CC(CO)C2)=O)ccc2oc(O)nc2c1 C1(N(C(COCc2ncc(C)o2)=O)C)CC2CCC(C1)N2C(C1CCC2CC12)=O N1(C(c2c(C(C)C)[nH]cc2)=O)CCC(CF)(NC(c2ncccc2F)=O)C1 c1(CC)nc(C)c(C(=O)NCC2CC(C(=O)NCc3cnn(C)c3C)C2)s1 c1(C(=O)NCCOCCCN(C(CCC=C=C)=O)C)ccc(C(C)=O)c(C)c1 c1nn(C)cc1Cl.N1(C(C)=O)CCN(CCCNC(C2(C3CC3)CC2)=O)CC1 N1(C(CS(=O)(=O)NC)=O)CCC2(CCCCC2NC(c2cccs2)=O)C1 C1(CC(=O)NCc2c(C)ccnc2)CCCN(C(=O)C(C)n2cccn2)CC1 C1(NC(C(C=C)(C)CC)=O)CCN(C(c2c[nH]c(=NCC)s2)=O)CC1(C)C C1(c2ccccc2)(C(N2CC(C)(NC(C3CCC(C)S3)=O)C2)=O)CC2(CC2)C1 C1(NC(C2N(CCCC)CCOC2)=O)CC2(CCN(C(=O)C3=CCCS3)C2)C1 N1(C(Cc2cc(C(C)C)no2)=O)CCC(CO)(NC(C2CC=CCC2C)=O)C1 c1(NCCC(=O)Sc2n(CC)c(-c3ccccc3C)nn2)cc(F)cc(F)c1 N1(C(C(=O)NC)=O)CC(O)(C2CCN(C(C3CCC(C)C3)=O)CC2)C1 C(=O)(C=C1SCC(=O)N1C)N1C(CNC(C(C)C2CCOC2)=O)CCCC1 N1(C(C(C)(C)F)=O)CC2CCC2(NC(c2ccc(-c3ccco3)nc2O)=O)C1 N1(C(=O)NCC(C)S(C)=O)CCc2c(Cl)cccc2C1 C(=O)(C1SCCc2ccccc21)NCC1(O)CN(C(C(C(C)C)CO)=O)C1 c1(CC)nccnc1C(=O)N(CC(C)NC(=O)CC1OCCO1)CC N1(c2cc(C)nc(C)n2)CCC2(CC1)CC=CC(=O)N2C c1(C(=O)NC2C(NC(c3csc(CO)n3)=O)COC2)csc(Cl)c1Cl n1(CC(=C)C)nnnc1CN(CC(C)CNC(C1CCC1(C)C)=O)C Cc1cccc(C(N2CCCC(N(C)C(c3cc(C)n(C)n3)=O)CC2)=O)c1F N1(CC(C2CNC2)OCC)CCc2cc(OC)c(OCC)cc2CCC1 c1(CC)c(C(=O)NC2CC2NC(c2cc(OC)c(Br)s2)=O)cnn1CC C1(C(C)C)CN(C(=O)C(F)(F)C2CC2)CCN1C(=O)Nc1cscn1 c1(NC)snc(C)c1C(=O)NCCC(C)N(C(=O)C=CC(C)(C)SC)C O=C(O)CC(c1cn(CCc2ccccn2)nn1)NC(=O)C(=O)NCC1CCC1 C(CC(C(=O)NCCC(O)C1CCC1)NC(c1nc(O)sc1C)=O)SC C1(NC(C2N(C(C)=O)CCCC2)=O)CC2(CCN(C(c3cc(CO)no3)=O)C2)C1 N1(C(C(=O)NCCc2ccc(Cl)s2)=O)C2CCC1CN(Cc1ccccn1)CC2 C1(C)(C(=O)NCC2C(NC(CC3C(C)C3(F)F)=O)CCC2)CC(C(C)(C)C)=NO1 Cc1ccc(F)c(NC(C2CCC(CNC(=O)CCC3CCCN3C)CC2)=O)c1 CC1(C)CC(CNC(c2sccc2-c2nn[nH]n2)=O)CNC1=O C1(C(=O)NOCC(C)(C)C)C2CCC(C2)C1CO.C=C1CCC(C(=O)N)CC1 O(C=C(C#N)C(=O)N1CCN(C(=O)C(c2ccc(C)s2)C)CC1C)CC N1(C(C(C(C)C)N2CCCCC2)=O)CCC2CCN(C(=O)CC3CC3)C2C1 c1(C(=O)NCC2(NC(C3C(c4cccc(C)c4)CC3)=O)CC2)cc(C)c(C)nn1 C=Cn1ncc(C(=O)NCC2CC2C(=O)NC2CC(O)CC2O)c1N Cc1ccccc1C=CC(N1CC2(C(=O)NC3CCCC3CO)CC1CO2)=O Cc1ncc(C(=O)NCC(C)CNC(C2CCN2Cc2ccccc2)=O)c(C)n1 c1(OCC(=O)NCCNC(c2nn(CC)nc2C)=O)cc(C)ccc1C N1(C(C(c2cccs2)NC(COCC)=O)=O)CCC1(C)CC C(CCC(C)C)(C(=O)NCC(C1CC1)N(C(c1cc(C)cs1)=O)CC)NC(=O)OC C1(C(=O)NCCCCC2CN(C(CC3CCC(C)(C)O3)=O)C2)CC2C=CC1C21CC1 C(=O)(C(COC)CC(C)C)N1CC2(N(C(C(C)SCCCC)=O)CC2)C1 CC(C)CC(F)(F)C(=O)NC(C1CCN(C(=O)COCc2ccccc2)C1)C C1(CC(=O)N(C2(C(=O)NC3CC4(CSC4)C3)CCC2)C2CC2)CCC(O)CC1 C(=O)(C1=CNC2=NCCC2=C1)N1CCCC(CCNC(Cc2nnc(C)o2)=O)C1 c1(C(N(C2CCN(C(C34CCC(OC)C3C4)=O)C2)C)=O)cc(N)c(F)c(F)c1Cl C1(NC(c2cncc(C)c2)=O)CN(Cc2cc(C3CC3)on2)CC(F)(F)C1 C1(C(=O)NCCC(C(=O)N2C(C(=O)OC)CC2)OC)CCOCC1(C)C N1(C(CC(C)OC)=O)CCCC(C)(NC(c2cccc(-n3cnnn3)c2)=O)C1 c1(C(=O)NCCC(C)NC(=O)CCC(C)(C)[N+](=O)[O-])cc2cc(Cl)cnc2o1 C12(C(N3C(COC)CC3)=O)CCCC1CCN2C(C1(O)CCCC1)=O N1(C(=O)CCC2CCC2)CCN(C(c2noc3c2CCCC3)=O)CC(O)C1 C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCC(NC(c2c(C)cc(=O)oc2C)=O)C1 Cc1ccc(NC(C2CCN(C(=O)C(C)C3CC3)CC2C)=O)c(C)c1 c1(C(=O)NC(CNC(c2c(C)coc2C)=O)(C)C2CCC2)ccc2c(c1)OCC2 c1(C(N(C(CNC(CCCOCCC)=O)C)CC)=O)n[nH]c2c(C)cccc12 C1(CC(N2CC(CC(C)NC(C3(C(=O)NC)CCC3)=O)C2)=O)CCCC(C)C1 c1(NC(C)=O)cc(C(=O)NC2CC3(C2)CC32CCC2)ccc1[N+](=O)[O-] C1(CNC(=O)Cn2ccccc2=O)C2CCC1CN(C(=O)CSc1nc[nH]n1)C2 C(CC(C(=O)NC(c1cnc(C)s1)C)NC(=O)Cc1cn(C)nc1C)OC c1(C2CCN(C(c3c(C)cc(F)cn3)C(=O)NC(C)C)C2)coc2ccccc12 c1(C(=O)NC(CC)CN(C(=O)C(c2cccc(F)c2)C)C)c(F)cc(F)cc1F N1(C(CC(=O)OC)=O)CCCC(C2CCCN(C(=O)CN3CCCC3)C2)C1 N1(C(c2ccc3nccn3n2)=O)CCC2CCN(C(c3cc(F)c[nH]3)=O)C2C1 Cc1c(C(=O)NC2CCC2NC(=O)CC2CC2)c(-c2ccccc2)cn1C c1(-c2cn(CC3N(C(C4CCNC4=O)=O)CCC3)nn2)c(F)cc(F)cc1F N1(C(C(=O)NCc2ncc(-c3cn(CC)nn3)o2)=O)CCCC(C)(CC)C1 N1(C(C(C)(C)SC)=O)CCCOC(CCNC(C2CC2F)=O)C1 C1(NC(c2nc(CC)oc2)=O)CCCC(C(=O)NCCCCN2CCC2)C1 c1(C(=O)NCC2C(NC(C3(O)CCC(CC)CC3)=O)C2)cc2ccc(C)cc2[nH]1 C1(C(N(CC(C)NC(=O)COCC(F)F)C)=O)COc2ccc(Cl)cc2O1 N1(C(CCCOCC)=O)CCN(C(=O)C(C)Sc2ccc(Cl)cc2)CC1C c1(NC(c2ccncn2)C)nc(N2CCN3C(=O)CCC3C2)nc2scnc12 c1(CC(=O)NCC2CN(C(=O)CC3CC3)CC2(F)F)c(F)cccc1Cl c1(C(=O)NCC2N(C(CC3(CSC)CC3)=O)CCCC2C)cc(C)c(C#N)cn1 C1(NC(c2c(C)nc(CO)s2)=O)CCN(C(C2CCC3CC3CC2)=O)CC1(C)C C1(C(=O)NCCC2(CNC(C3(C)CCC4CC4C3)=O)CC2)CN=C2N=CNN2C1 C1(NC(=O)C2=COCCC2)COC2(CCCN(C(=O)COCC3CCCC3)C2)C1 C12(NN3CCC(C(=O)OC(C)(C)C)C3=O)CCC(C1)N(C(=O)C(O)C(C)(C)C)C2 CC(c1ccc(F)cc1)=CC(=O)NCC1C(C)CCCN1C(c1cncnc1)=O C1(CNC(C(C)OCC(F)(F)F)=O)CN(C)CCN1C(c1cc2[nH]ccc2s1)=O C(=O)(CC(F)(F)c1ncccc1Br)N(CCOCC)C.n12cc(nn1)SCC2 C(=O)(C(C)Cc1ccc(CC)o1)NC1CN(C(CCOCC#C)=O)C1 N1(C(C2CC(SC)C2)=O)C2CCCC1CC(NC(=O)C(C(C)C)C(C)C)C2 c1(C(=O)NCCC2CC(NC(=O)CC=C(Cl)Cl)C2)cccc(C#CCO)c1 C1(C(=O)NCC2CCN(C(C3(COCC)CC3)=O)C2)CC12C1CC3CC(C1)CC2C3 c1(CO)cnn(CCO)c1.C1(OCCn2c(C3(C)CO3)nnn2)COC(=O)C1 N1(C(CCOc2cc(C(C)=O)ncc2)=O)CC2CC(CO)(C2)C1 Cc1cc2c(cc1C)OC(C(=O)NC(C)CCNC(c1cc(C)c(N)cn1)=O)C2 c1(N(C)C)nc2ccc(COC(=O)CC3CCCC3(F)F)cc2o1 N1(C(c2c(COC)noc2)=O)CCC2(CC2C(=O)NC2C=CCCC2)C1 CC1=C(C(=O)N2CC(CO)(NC(c3snnc3C(C)C)=O)C2)C(=O)OC1(C)C c1(C(N2CC(N(C)Cc3cccc(S(C)=O)c3)C2)=O)ncnc2[nH]cc(I)c12 CC1=CCC(C(N2CC3CC3C2CNC(=O)Cc2cnc[nH]2)=O)CC1 Cn1ncc2ncnc(NC3CC(CC(=O)NCCOC4CCCC4)C3)c12 c1(C(=O)NC2CN(C(c3c(OC)n[nH]c3)=O)CC2O)cnc2cc(C)nn2c1C c1(C(c2nnnn2C(OCCNC=O)C2CC2)CN)csc(C2CCCO2)n1.C1CC1 N1(C(C(CCNC(=O)CCC(C)CN(C)C)OC)=O)CC2CCN(C)C2C1 c1(C(C)NC(C2N(C(C=C(C)C(C)C)=O)CCC2)=O)c(C)noc1C Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CCCNC(N)=O)nn1C C12(C(=O)NCC=C3CCN(C(C(C(C)OC)O)=O)CC3)CC(C)(C1)OC21CCC1 CC1(C)C(NC(=O)NCc2cc(N3CCCC3)ccn2)CC1C(F)(F)F C12(CNC(COCC)=O)CCC1CN(C(c1cccc(NC3CC3)c1)=O)C2 C=CC(O)C(=O)N1CCC(C2CCCN2C(=O)C=CCN(CC)CC)C1 C1(CCNC(C(C)OCCCC)=O)CCCCN1C(C1CCC(C(N)=O)CC1)=O N1(C(C(=O)Nc2cccc(-c3nc(C)[nH]n3)c2)=O)CCC(C2(O)CC2)CC1 C(CC(CC)C(=O)NCCCOCCNC(=O)CC1(C)CCOCC1)=CC Cc1cc(Br)c(NC(c2cnc(C(F)F)cn2)=O)cc1Cl C1(C(N(C2CN(C(c3cc(C)sc3)=O)CC2F)C)=O)CC(C)CCC1C(C)C C1(C(N2CC(CNC(C(C)OCCC(C)C)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 N1(C(c2cc(C)no2)=O)CCC12CC(C(=O)NC1C3CC4C(C3)C14)C2 c1(C(N2CC(C(=O)OC)C(OC)C2)=O)cc2c(nc1Cl)COCC2 C1(C(=O)NCC(C)NC(C2(OC3CCOCC3)CC2)=O)OCC1(C)C c1(C(=O)NCC(=O)NC2CC(NC(CC3(C(=O)NC)CCC3)=O)C2)ccccc1 Cc1ccc(Cl)cc1OCCCC(=O)N1CCC(CNC(=O)C2=NOC(C)C2)C1 c1(CNC(C2(CC=C)CCC2)=O)cc[nH]c1C(=O)N(CC(O)C1CC1)C c1(CC)cc(F)ccc1CC(=O)NCC1CCC1NC(=O)C=C(C)c1ccsc1 c1(C(=O)NCC2OCCC3CN(C(CNC(C)=O)=O)CC32)cc(C)nc2ccnn12 c1(C(N2CCCC(NC(c3c(=N)cc[nH]c3)=O)C2)=O)cnn2c1OCC(F)C2 C1(CNC(=O)CN2CSCC2=O)CC(C(=O)NCCOc2ccncc2)=NO1 C(=O)(C1=CCCSC1)NC1(CCNC(C2(C)CS(=O)(=O)C2)=O)CC1 c1(-c2cn(-c3c(C)n(-c4ccccc4Cl)nc3)nn2)cccc2cccnc12 CCC(CN(C)C)C(=O)N1CCC(CC(=O)N(C(C)COCC)C(C)C)CC1 CC1CC(=O)NCC1C(N1CC(C)(C(=O)NCCSC(C)(C)C)C1)=O N1(C(C(C)(C)C)=O)CCN(C(=O)CN2CCN(C(C3CCC3(F)F)=O)CC2)CC1 c1(C(N2CC(N(C(c3c(C)cc[nH]3)=O)C)C(O)C2)=O)ncc(N)cc1C c1(N(C)C)ccc(C(c2nnnn2C2CCC2)NC2CONC2=O)cn1 Cc1cc(C#N)cnc1C(=O)NC12CCN(C(c3ccc(CO)o3)=O)CC1C2 C(=O)(C(CC(C)C)OC1CCCC1)C(C)OCC(=O)NCCN(C(=O)CCOC)C c1(C(F)(F)F)c[nH]c2cc(F)c(F)c(F)c12.c1(C2CN2)cccc(Cl)c1 C(N=c1[nH]c(=N)[nH]c(=NCC2(C)CCC(F)(F)CC2)[nH]1)C1CCCC(CC)CC1 N1(C(C2(OCC)CCCC2)=O)CC(NC(=O)CC2(C)CC2(F)F)C(C)C1 C(=O)(CCCCC(=O)NC1C=CC(CNC(=O)Cc2c(C)nn(C)c2C)C1)OC c1(OC)cc(F)c(C(=O)N(CCCNC(c2ccnc(CO)c2)=O)C)c(F)c1F C#CCC(C(=O)NCC(=O)OC)NC(c1csnn1)=O N1(C(CNC(=O)NCc2cccc(N)c2)=O)CCN(C(=O)CC2CC2)C2CC12 N1(C(c2c(CCC)[nH]cc2)=O)CCCC2(CCC(NC(=O)C=C(CC)CC)C2)C1 CC1c2ccccc2OC1C(=O)NCC1(C)CCN(C(=O)CCC#N)CC1 C1(C(=O)NCC2(COC)CN(C(=O)C3=COCCC3)C2)CCn2c(C)cnc2C1 c1(C(N2CCCC2CC(N)=O)C(=O)NC2(C)CC2)cnc(C2CC2)o1 C(N=c1[nH]c2cc(Br)ccc2o1)C1CCN(S(=O)(=O)c2cccc(Br)n2)C1 c1(C(=O)NC2C(NC(c3cc(C)on3)=O)CC2)cc(C(C)(F)F)ccc1C C(=O)(C1=CC2C=CC1C2)NC1CCC(CCNC(c2c(C)nncc2)=O)C1 C=C(C)CCCC(=O)NC1CC=C(C(=O)NC(C)(C)COC)C1 C1(NC(=O)C=CC2CCCC2)CN(C(=O)COCC(F)F)CC12CC2 N1(C(=O)CCc2nc[nH]n2)CCC2(CCCN2C(c2cc(=O)cc(Cl)[nH]2)=O)C1 C(CC(CC)C(=O)N(CC(=O)NCCc1cc(C)no1)CC1CCC1)=CC N1(C(C(C)=C2CC2)=O)CCOCC(NC(c2cnnn2C2CC2)=O)C1 CC1(NC(C23CCCC2C3(F)F)=O)CCCN(C(=O)C=Cc2ccccc2)C1 C1(NC(C=CCC(C)(C)NC(=O)C=Cc2ccncc2)=O)CCC2CC1CO2 N1(C(CSC(c2ccccc2)C)=O)CC(N(C(=O)CC2CC=CC2)C)C(O)C1 C1(CC(=O)NCCCOCC(C)C)C2CCCC2N1C(C1CCOC1C)=O N1(C(CC(CC)OC)=O)C2CCC1CC(C(=O)NC(C)C(F)(F)F)C2 C12(NC(CS(=O)(=O)NC)=O)CCOCC1CN(C(c1ccc(C#N)cn1)=O)C2 C1(C#N)(C(=O)NCCCNC(CCN(C)CC)=O)CC2CC2C1 n1(CC)cnnc1C1CC1C(=O)NCCN(C(=O)C(F)CC1CCCCC1)CC c12cccc(c1)OCC(=O)N1CC(C1)C(C)NC2=O.n1(CC)cc(NC)cn1 c1(CC)cc(C(=O)N(C(C)C(=O)NC2CC(n3cccn3)C2)CC)n[nH]1 C1(C(N2CC(C)CC(NC(c3c(C)ccs3)=O)C2)=O)CC2CCCC(C1)C2=O C(=O)(C(C#N)C(C)(C)C)NCC(C)(C)OCCNC(CCC(C)OC)=O C1(NC(C=CC(=O)NCCC(C)N(C(=O)C(F)CN(C)C)C)=O)CCOCC1 C=C(C)C1OCCCC1C(=O)NC1CN(C(c2ccnnc2C)=O)CC1O c1(C(N2C(CN(C(CC(CC)OC)=O)C)COCC2)=O)c(N)sc(C)c1C CC(C)C(C(C)NCc1cnn(C2CC2)c1)NC(=O)Cn1ccc(C2CC2)n1 c1(C(N(CCNC(C(c2c(C)cccn2)(F)F)=O)C)=O)cc2c(nn1)CCCO2 CCC(CN(C)C)CC(=O)NCC1(F)CCN(C(c2ocnc2C(F)F)=O)CC1 C(C1CN2CC1C2=O)=CC(=O)NCC(C)N(C)C(C)=O.C1(SC)CCCC1 c1(-c2nnc(N(NS(N)(=O)=O)CC)n2CC(=O)N(C)C)ccc(OC)c(OC)c1 CN(C)S(=O)(=O)N1CCN(C(C)N2CCCCC2)C1 c1(C(C)C)ccc(O)c(C(N2CC3CC3(NC(c3ccc(F)c(F)c3)=O)C2)=O)c1 c1(CC(N2CC(C(C)NC(=O)Cn3cnc(Br)c3)C2)=O)ccc(OCCF)cn1 N1(C(CC(CNC(c2c(C)cccc2F)=O)C2CCC2)=O)CCN2CCC1CC2 CC(N=c1nc2c(cnn2C)c(N(C2CC3(CC3)C2)C2CC2)[nH]1)c1ccc(Cl)cc1F C#CCC(C(=O)N1CCC1)NC(=O)CCc1ccncc1.c1sccc1Cl S(=O)(=O)(c1ccncc1)N1CC(F)CC(C(=O)Nc2cc(C)c(F)cc2)C1 c1(C(N2CC(C)(NC(c3cc(C(C)=O)on3)=O)C2)=O)ccc(SC2CCC2)cc1 CC1(C)CC(NC(c2ccc(CO)c(F)c2)=O)CN1C(c1cc(F)c[nH]1)=O CCCCC(O)CC(=O)NC(CN(C(C1COCCN1CC(F)F)=O)CC)CC C(=O)(C1=NOCC1)NCC=CCC(=O)N(C)Cc1cn(C)cn1 C(=O)(CCCCCCCCCCCC)NCCC(=C)CNC(=O)CCC(C)(F)F CC(C(=O)NCC1(CNC(=O)CCCc2ccccc2)CC1)C(F)F C1(C(=O)NCc2cn(C(C)C)nn2)CCCCC1OC(c1cccc(Cl)c1)=O C(=O)(CC1=CCOCC1)NCC(C(C)C)NC(c1ncoc1-c1ccco1)=O N1(C(C(CC)OC)=O)CCC(O)(C(C)NC(c2snc(O)c2Cl)=O)CC1 C(=O)(CCCCCCNC(=O)C(F)C(C)C)N(CC(CC)CC)CCO N1(Cc2cnc(OC)nc2)CCN(C(=O)C(Cl)(Cl)Cl)C2CC12 c1(C(=O)NC(C)CNC(c2cscc2C(F)(F)F)=O)ccnc2[nH]ncc12 C=CCCCCCC(=O)NC1CC(C)(NC(=O)Cc2csc(C(F)(F)F)n2)C1 N1(C(C(CCC)OC)=O)CC2CC(C1)N(C(=O)C1CC1)C2.O(C)OC.OC N1(C(c2csnn2)=O)CCCC1Cc1cn(-c2cnsn2)nn1 C(C(CC)CCC)(c1nnnn1C)NC1CC(=O)N(CCC)C1=O C(=O)(NNC(=O)C(=O)NCS(=O)(=O)C(C)(C)C)c1ccc(OC)cc1 C1(NC(c2cccc(N(C)C)n2)=O)CCCN(C(c2c(I)cnn2C)=O)CC1 c1(C(N(CC(C)CNC(C2CCC23CCC3)=O)C)=O)cc2c([nH]1)CCCC2 c1(CS(=O)(=O)NC)ccc(CNC(c2sccc2Nc2ncc(C)cn2)=O)cc1 S(=O)(=O)(c1cccs1)NC(C(=O)NCC(CC(F)(F)F)NC(CC(C)CF)=O)C C(=O)(C(F)CCC(C)(C)C)N1CC2(C(NC(C(CCC)F)=O)CCC2)C1 C(=O)(C(C)(C)CCCNC(c1ccc(C(N)=O)[nH]1)=O)NCCc1cnc(C)[nH]1 C1(C(N2OCC(n3cc(CNC(N)=O)nn3)C2)=O)CC12CCS(=O)(=O)CC2 C1(NC(=O)NCCCC)CCCN(C(c2c(C)noc2CC)=O)CC1 Cc1cc(CCC(=O)NCC2CN(C(c3cnc(C(N)=O)cn3)=O)C2)cc(C)n1 C1(C(=O)NC23CC(CNC(C4N(C)CC4)=O)(C2)C3)CCCC1C1CC1 Cc1c(C(N2CCCC(c3ccncc3)CC2)=O)cc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(C(C)NC=O)=O)CCC(C(=O)NCCS(C)(=O)=O)(CO)C1 N#Cc1cc(CN2CCC(O)(CO)CC2)cc(-c2ccc(Cl)cc2)c1 CCCC(C)(O)CC(=O)NC1(CNC(C2(O)CCC(C)(C)CC2)=O)CCOCC1 C(=O)(CCCCCCCC1CC1)N1CCC(Nc2nccc(OCC)n2)C(C)C1 c1(C(N2C(C)CCC(NC(c3cnc(CC)s3)=O)C2)=O)cnc2[nH]c(O)nc2c1 C1(OC)CC2(C1)CN(C(=O)C(CC(N)=O)NC(c1csc(F)c1)=O)C2 C1(NC(CC=CC=C)=O)CCN(C(c2cnc(C(F)F)c(C)c2)=O)CC1C CCCC(CCC)C(C)(c1nnnn1CCC1CC1)NC1CC2CC2C1 c1(C(c2n(CCOC)nnn2)NC2CCCC2)ccc(OC)c(OC)c1 c1(NC(=O)NC(CC(CC)C)C)c2c(nn1C)CN(C(=O)OC(C)(C)C)C2 C12(NC(c3cc[nH]n3)=O)CN(C(c3c[nH]cc(F)c3=O)=O)CC1CS(=O)(=O)C2 C(C1=CCN(C)CC1)NC(C1CCCN(C(CCn2c(C)ncc2)=O)C1)=O C(CC(F)(F)C(F)(F)Br)(C(=O)O)NCc1cccc2nnn(C)c21 c1(C(N(C2CCN(C(c3cnc(Cl)[nH]3)=O)C2)CC)=O)cnc(C(C)OC)s1 C=C(C)CCCC(=O)N1CCN(C(c2cc(C(F)(F)F)cc(F)c2)=O)CC1C CC1CCc2n[nH]cc2C1C(=O)NCC1CC(NC(c2ccc[n+]([O-])c2)=O)C1 c1(C(=O)NC)ccc2cc[nH]c2c1.C(=O)(C1C(C)N1)NCC1CCN(C(C)=O)C1 C1(COC(CC(C)(C)OC)=O)CCn2ccnc2C1 N1(C(C(CC)C(=O)OC)=O)CC(O)CCC1C(N1CC(O)C(O)C1CO)=O c1(NC(C(c2cc(C)cc(Br)c2)N2CCC(O)C2(C)C)=O)ccc2c(c1)OCO2 C1(F)(CNC(CC2CN(C)C2)=O)CCC(NC(=O)CCSCc2ccccn2)C1 Cc1ccc(CCC(=O)NC(C)(CNC(=O)Cc2ccc(Cl)cc2)CO)cc1C N1(C(c2c(OC)nc(C)cc2)=O)CCC2CCCN(C(C3CN(C)C3)=O)C2C1 Cc1ccc(SCCC(=O)NCC(=O)OC(=O)CCc2cnc(O)[nH]2)cc1.C1C(F)C1 C(C(=O)NCC(CCNC(=O)CNC(c1ccccc1)=O)OC)(C(C)C)SC N#Cc1c[nH]c2ncnc(N3CCC(NC(=O)CCN4CCOCC4)C(O)C3)c12 CCC(F)(C(=O)OC)C(=O)NCC(C)CNC(C1(Sc2ccccc2)CC1)=O c1(C(=O)NCCOCCOCCNC(C2(F)CCCC2)=O)nccc2nn[nH]c12 C1(CNC(CC(=C)C)=O)CC2CCC1N(C(C1CC=C(C)CC1)=O)C2 N1(C(C(CC)C(=O)OC)=O)CCOC2CN(C(c3cc(C(F)(F)F)[nH]c3C)=O)CC12 c1(SC(C(N2CC(NC(C(CCCC)O)=O)(CO)C2)=O)C)nc2ccccc2s1 S(=O)(=O)(c1nc(N2CC3CCC(O)C3C2)ccc1Br)N(C)C c1(C(N2CCCC(CNC(C3CC(CC)C3)=O)C2)=O)cnc2c(c1)NC(=O)CS2 C(=O)(CS(=O)(=O)CCO)N(CC(C)NC(=O)CC1CC(C)=NO1)CC C12(NC(CCCC#C)=O)CN(C(=O)CN3CCN(C)C3=O)CC1CS(=O)(=O)C2 c1(C2(C)C(N(CCOCCN(CCC3CC3)CC)C)C2)ccccc1 N1(C(C(C)S)=O)CC2CN(C(c3cccc(N4CCOCC4)c3)=O)C2C1 C(C(C)(O)CC(=O)N1CC(n2cc(-c3ccc(OC)s3)nn2)C(C)C1)OC c1(C(=O)NCC(=O)NCC2CC(OC)C2(C)C)ccc2occc2c1 C1(OC(c2scc(C(=O)NCC3CCN3C(=O)COC)n2)(C)C)CCCCCC1 c1(OC)cc(C(N2CC(OC)C(NC(=O)CCNC3CCC3)C2)=O)cc(N)c1O C(CC(C(=O)NCC1C(C)(C)C1(C)C)NC(=O)CC(C)(C)C1CCCC1)N(C)C c1(CC)nsc(NC2CC2)n1.c12cnn(c1)[nH]c(=O)c2=O.C12CC1CNC2=O c1(NC(C2N(Cc3sc(C)c(Br)c3)CC2)=O)nc2ccc(F)cn2n1 c1(OC)nc(N2CC3CC(NC(C4COC(C)C4)=O)CC2C3)nc(C)c1F c1(C(N(C(CNC(C(C(CC)C)C)=O)C2CC2)C)=O)cccc2c1CCCC2 N1(C(C(C)(C)C(F)(F)F)=O)CCOC2(CCN(C(=O)C=C3CC3)C2)C1 C1(C(=O)NC2C(C)CN(C(C3CCC(=O)N(C4CC4)C3)=O)C2)CCC(F)(F)CC1 c1(C(N2CC(NC(CNC(CC)=O)=O)CC3(C2)CC3)=O)nnc2ccccc2n1 C1(C(N2C(COC)C=CCC2)=O)CN(C(C2CCC(O)CN2C)=O)CCN1C c1(C(=O)NC23CC(NC(c4ccn(C(C)C)n4)=O)(C2)C3)ccc(Br)c([N+](=O)[O-])c1 Cc1nn(C)cc1CCC(=O)N(C1C2CN(C(=O)CNC(=O)NC3CC3)CC12)C C1(C(=O)NCC2N(C(c3c(C)cco3)=O)CCC2)CC12CC(C)(C)C2 C(CC(C(=O)NC1(C(F)(F)F)CC1)NC(=O)C(C1CCCCC1)OC)=CC c1(C(=O)NCC2(NC(c3cc[nH]n3)=O)CCC2)cnn2ccncc12 N1(CCNC(c2c(C)onc2)=O)CCC(NC(c2ocnc2C(F)F)=O)CC1 N1(C(=O)NCC2(c3ccccc3)CC(O)C2)CC2(CCCCC2)C1c1ccccc1 N1(C(Cn2c(C)ccn2)=O)CCC(C(=O)NC(C)Cc2nncn2C)C1C CC(C)C(F)C(=O)NC1(CNC(c2ccc(NC=O)cc2)=O)CCOC1 Cc1cccc(C(=O)NCCC2(O)CN(C(=O)C(O)CN3CCOCC3)C2)c1F c1(C(N(CC(C)(C)NC(=O)Cn2nc(O)ccc2=O)C)=O)cc2n(c1)CCOC2 c1(C(N2C(CN(c3n[nH]c4c3CCC4)CC)CCC2)=O)cc(OC)cc(Cl)c1 N1(C(c2cc(C)nc(Cl)c2)=O)CCOC2(CCN(C(=O)C(F)(F)C(F)F)CC2)C1 CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cncc(C)c3Cl)=O)C2)CC1 N1(C(C2(C)CC(C)OCC2)=O)CC2CCCC2(NC(c2cnco2)=O)C1 c1(C(=O)NC(C2CCN(Cc3cc[nH]c3)CC2)C)ccc2nc(Br)sc2c1 C#Cc1cc(C(N2CC(NC(=O)CCS(C)(=O)=O)CC(C(F)(F)F)C2)=O)ccc1C c1(NCc2c(COC)ocn2)cc(NCC2CN(C)CCN2C)nc(C)n1 C(=O)(CC1=CCOCC1)NC(C(C)NC(CCc1cccc(C(=O)NC)c1)=O)C c1(OCC)cnc(C(N2CCC(CO)(NC(=O)CC3CCC(=O)NC3)C2)=O)cn1 c1(C2(C(=O)NC(C(=O)NC)CC3CCCO3)CC2)ccccc1Cl.N1(C)CCCCC1 c1(SC)cccc(C(=O)NCCOC2CCN(C(c3cc(Cl)n(C)n3)=O)CC2)c1 CCC(CCOC)C(=O)NC1CCCCCC1C(=O)NC(CN1CCCC1)CO c1(C(=O)NCCCCCNC(Cn2c(CCC)ncc2)=O)ncc(Cl)cc1Cl C(=O)(CCCC(F)(F)CO)NC(C)C(C)(C)NC(C1CCS(=O)(=O)CC1)=O C(=O)(CC1=CCOCC1)NC1C(Cc2cn(C3C(C)(C)SCC3)nn2)C1 c1(NC2CC(C)OCC2)ccccc1S(=O)(=O)CC(=O)OC(C)(C)C C1(C(=O)NCC(CCCC)O)CC2CN(C(=O)CC(F)(F)F)CC2C1 CSC1=C(C(=O)NC2C3CC4C2C4C3NC(C2CN3CCCN2CC3)=O)CCCC1 C(=O)(C1=CCC(NC(C2C=CCCC2)=O)C1)NCc1n(C(C)C)cnc1 c1(C(C(=O)NC(CC)C)N(C2CC3CC2C2CC32)C)cc2occc2s1 CCC(CC(=O)NCC(C)N(C)C(C1CCCC1O)=O)c1ccccc1 C1(C(=O)NC2(COC)CC2)CCC2(CC2)N1C(c1cc(CO)nn1C)=O CCCN=C(NCCOc1cccc(SC(F)(F)F)c1)NCC(C)(C)CN(C)C c1(CC(=O)NCCNC(C(c2ccccc2)C)=O)cncn1C.C1CC(C)(C)C1 c1(N2CC3CC(NC(C4C(=C)C4)=O)CC3C2)cc2nnc(C(C)(C)C)n2cn1 CC1CC(c2nnnn2CC2CC2)(NCCCSc2ccccc2)CN1C C1(NC(Cc2cn(CC)nc2)=O)CC2CCC1N(C(=O)C(N1CCNC1=O)C)C2 c1(CNC(CC(OC)OC)(C)c2nnnn2C)sc2ccccc2c1CS(C)=O C1(C(=O)NCC2CN(c3ccnc(C(CC)C)n3)C(C)C2)CC(=O)CC12CCC2 n1(CC(=O)NCC(CC)NC(C2(C(F)F)CCC2)=O)nc(O)ccc1=O N1(C(c2c(CC)cccn2)=O)CC(CC(=O)NCCC(C(C)C)N(C)C)C2(CC2)C1 c1(NC(CC2CC(OC)C2)=O)cnccc1C(=O)NC1CC(=O)NC1=O c1(C2(C(N3CC(O)(CNC(C4(CO)CC4)=O)C3)=O)CC2)cccc2ccccc12 c1(CN2CC3C(NC(c4ncc(C)nc4)=O)C3C2)cc(Cl)c(O)c(Br)c1 C1(C)(CNC(C)=O)CN(Cc2ccccc2)CCO1.C12COCCC1C(=O)N2 C1(C(=O)NC(CC2CC2)C(N2CCN(CC3CC3)CC2)=O)CC2(CCCCC2)C1 C(=O)(C(=O)CC(C)C)N(CCCNC(CCC(=O)NCCC)=O)CC C(=O)(CC(CC)C(F)F)N1CC(C(=O)NCC=CC)C(CCC)C1 Cc1cncc(-c2cn(C(C)C(=O)NCCc3ccc(C(=O)O)cc3)nn2)c1 C12(NC(c3c(C)coc3C)=O)CC3CCC(C1C2)N3C(c1cc(CCO)on1)=O N1(C(c2c(N)sc(C)c2C)=O)CCCCC(NC(=O)C(N2CCSCC2)C)CC1 O=C(CONC(=O)C1CCSC1)N1Cc2ccccc2CO1 C(CN=c1[nH]c(C2CCCCC2)nc(=N)[nH]1)N(C(C1CC(C)OC1)=O)CCO C1(C(=O)NCC(C)OCCO)C2CCC(C2)N1C(c1c[nH]c(=N)o1)=O C1(C(=O)NC(CC)CNC(c2cc(CC3CC3)on2)=O)CCCC1(C)C N1(C(C2C(C)(C)C2(C)C)=O)CC2CCC(CNC(=O)CC(F)(F)Cl)C2C1 N1(C(C(CC(C)C)NC(C)=O)=O)CCC2(C1)CN(C(=O)CCC(=O)OC(C)(C)C)C2 C(=O)(CCC(O)C(C)(C)C)N1CC2CC(NC(C3C(C)(C)CO3)=O)CC2C1 N1(C(c2nc(C)c(C)[nH]2)=O)CCCC(CCNC(c2ccncc2F)=O)CC1 C12(NC(C(CC)NC)=O)CCC(NC(=O)C(C)Oc3ccc(Cl)cc3)(CC1)C2 N1(C(C(C2CC(F)(F)C2)OC)=O)CCC(CN(C(=O)CC2CC=CC2)C)C1 c1(CC2N(C(=O)Nc3ccnn3-c3ccccc3)CC=C2)ccc(F)c(Br)c1 c1(C2C(C(NOCCC(=O)O)=O)C2)cncc(Cl)c1Cl Cc1ccc(CNC(C2CC23CC(NC(=O)Cc2csc(C)n2)C3)=O)cc1 C12(C(=O)NC3CCC(CNC(COCP(C)(C)=O)=O)C3)CCC(CC1)O2 C1(CNC(C(C=C)(C)O)=O)N(C(=O)Cc2ncc(Cl)s2)CCCC1(C)C N1(c2cc(C(=O)NCC(C)C)[nH]n2)CCN(C(C2CCC(Cl)CC2)=O)CC1 C1(C(N2CC(CCCCNC(Cc3ccc(C)s3)=O)C2)=O)CCOC(=O)CC1 c1(C(N(CC(C)NC(CNC(CCC)=O)=O)C)=O)cc(F)c(F)c(C#N)c1 c1(CCC)ccc(C(=O)N(C)CC2(CNC(=O)C(C)(C)OC)CC2)c(OC)c1 N(C(=NCCCCN1CCCC1)N1CCC(n2cccn2)C1)CCOC(C)C c1(CC(=O)NCC2C(CNC(COCC)=O)C2)cccc(O)c1F N1(C(c2cccc(N)c2)=O)CCC2(CNC(=O)CCN3CCCC3)CCCC12 C(=O)(C(F)CC1CN(C(=O)C(C2CCCCC2)O)C1)NCC=C(C)C n1(CCC)nc(C)c(C(=O)NC2CN(C(c3cncnc3CC)=O)CC2C)c1C C1(NC(CC(=O)OCC)=O)CN(C(=O)CCNS(C)(=O)=O)CC1C c1(OC)ccc(CO)cc1.c12sc(nc1C)[nH]c2=O c1(CC)cc(C(=O)NCC23CCCN(C(c4ncn(C)n4)=O)C2C3)c(C)nn1 c1(C(=O)NC2CC(CCNC(Cc3c(CC)con3)=O)C2)cc2ccccn2c1 Cc1cc2ccc(C(N3CCC(O)(C(C)CNC(=O)CCC(N)=O)C3)=O)cn2c1 C1(C)(C(=O)OC)CCN1C(c1ccc(CNC(=O)Cc2n[nH]c(C)n2)o1)=O CC(CN(C)C)CC(=O)NCCC1(O)CCN(C(=O)Cc2ccn(C)n2)C1 c1(C(=O)NC2CCN(C(CC(C)(C)C)=O)CC2F)cccc2c1CCCCC2 Cc1scnc1C(=O)NC(C)C(C)NC(=O)CN1CCC1C C(C1COC(C)(C)O1)=CC(=O)NC(C1CN(C(C2(F)CCOCC2)=O)CCO1)C N1(C(CCC#C)=O)CCCC12CCCN(C(C1(OC)CC(C)C1)=O)C2 C(=O)(CC(C)C(F)F)N(C1CCCN(C(C2C(C(C)=O)C2(C)C)=O)C1)CC1CC1 c1(C(=O)NCC(C)CNC(C2CCCC2C(F)F)=O)ccc2c(c1)NC(=O)CC2 c1(NCC(C)(C)C(F)(F)F)nc2ccccc2nc1NCc1ccc(F)cc1Cl Cc1ccc2c(c1)CCC(C(=O)NCC(C)NC(=O)CC1CC=CCC1)O2 C(=O)(CN=c1[nH]c(N2CCC(CN(C)C)C2)nc(=NC)[nH]1)NCC C1(N(C(CC(C=C)C)=O)C)CN(C(C2CC2CC(C)C)=O)CCC1O c1(OC)ccccc1-c1oncc1C(=O)N(CC(C)N(C(=O)C(C)N(C)C)C)C CC1CCN2CCCC2CN1c1cc(NCC2(CO)CC2)ncn1 c1(CC(=O)NC2C(CC)CN(C(C3CC3(C)CC)=O)C2)ccc(C#N)nc1 N1(C(CC(CNC(C(C)OCCOC)=O)C)=O)CCC2(COC(=O)N2)C1 N1(C(C(CC(C)C)O)=O)CC2(CCCCN2C(C2CCCC2O)=O)C1 c1(NC(=O)N(C2CC2)CC2CC23CC3(F)F)cccc(F)c1F C(CC(C)C)(C(=O)N1CCC(C(=O)NCC2(OC(C)C)CCC2)CC1C)OC C#Cc1ccc(C(N2CCCC2C(C)(C)C(=O)NCC2CCC2C)=O)cc1 Cc1nnc(-c2noc(CS(=O)CC3CCOCC3)n2)n1-c1ccccc1 c1(C(N2C(CCNC(CCC(C)SC)=O)COCC2)=O)coc2ccc(Cl)cc12 C1(C(=O)NCC2N(C(=O)CC(F)(F)F)CCC2)CN(C(=O)CO)C2(CCC2)C1 O(NC(=O)C(CNC(=O)C(C1CCCC1)OC)C(C)(C)C)CCCCC C1(CN(C(=O)CC2(C)CCN(C(=O)CCCCN(C)C)C2)C)OCCC1(C)C Cn1c(O)nc2cccc(C(N3C(CNC(c4cnn[nH]4)=O)CC4CC34)=O)c12 C(CC(=O)NC(c1snnc1C)C)(C(F)(F)F)NC(c1ccn(CCC)n1)=O c1(N(CC(C)NC(C2CCOC(C)C2)=O)C)ncc(C#N)cc1F C1(O)(CNC(c2cc(F)cs2)=O)CCCN(C(=O)C=Cc2cnc[nH]2)CC1 N1(C(c2n(C)nnc2)=O)CCC(C(N2CCOC3CC23)=O)CC1(C)C N1(c2ncc(-c3ccc(C)cc3)s2)CCC(F)C(NC(c2ccccc2)C)C1 Cc1nc(-n2nc(Cc3cnn(C)c3)nc2-c2cnn(CC(C)C)c2C)n(C)n1 CON1CCC(C(=O)NCCCN(C)C(C2CCC(C3CC3)C2)=O)CC1 C1(NC(COc2ccc(C)cc2C)=O)COC2(CCN(C(=O)C=CBr)CC2)C1 N1(C(C2(CC)CCCCC2)=O)CCC2(CCCN2C(=O)CC2CC(=O)NC2=O)C1 C1(CNC(C2(COC)CC2)=O)CC2CC(C1)N(C(=O)C(C)=C1CCC1)C2 c1(CCC)ccc(C(N2CCC(N(C)C(c3sncc3C)=O)C2)=O)cc1N C1(C(N2CCC(CN(C)C(C3CCCNS3(=O)=O)=O)C2)=O)CC2(COC(=O)N2)C1 C1(C(=O)NC2C3CCN(C(c4ccc(C)c(C)n4)=O)C32)CCCC(F)(F)CC1 c1(C(N2C3CCC2CN(C(C2CC2C2CC2)=O)C3)=O)ccc(F)c(F)c1Br C1(C(N2CCCC(C(=O)NCCc3cn[nH]c3)C2)=O)OCC2CCCC12 C(=O)(C(CC)C(=O)NCc1ccoc1C(=O)NCc1nn(C)c(=O)o1)OCC CN1CCN(C(C2CCC3(CC2)CC3)=O)CC1CNC(=O)CCF c1(CC)cccc(C(N2CCCC2C(C)CC)C(=O)NCCC#N)n1 N1(C(CCc2cn(CCCCC(=O)O)nn2)=O)CCC2(CCCO2)CC1 N1(C(C(C)C2CCCC2)=O)CC(NC(=O)Cn2ccnn2)C2(CC2)C1 C1(CNC(CC2(O)CC(C)(C)OC2)=O)CC2(CCN(C(C3(C)CCC3)=O)CC2)C1 CC(C)CC(O)CC(=O)NC1CCN(C(=O)Cc2cc(Cl)cc(Cl)c2)C1 c1(OC)nc(=NCC2CN(C(c3occc3C)=O)CC2C(F)(F)F)[nH]c(C)c1F N1(C(C2(C)CC(C)C2)=O)CCC(OCCCNC(C2CCC(N(C)C)C2)=O)CC1 C1(C)(C(=O)NC(C(c2cccc(CO)c2)C)=O)CN(c2nnc(CO)s2)CCO1 c1(CN(C2CCN(C(C3(C(C)C)CCC3)=O)C2)C(=O)CC2CC2)ccc(F)cc1 c1(C(=O)NC2CC(CCNC(C3(C)CS(=O)(=O)C3)=O)C2)cccc2[nH]c(=N)oc12 c1(OCC)ccc(C(=O)NC2(C)CCCN(C(=O)C(C)C3CCC3)C2)c(F)c1F c1(CCCC(N2CCC(CCNC(C(F)OC)=O)CC2)=O)nc2ccccc2o1 c1(C(N(C)CC2COCCN2C(=O)Cc2nccn2C)=O)nn(C)c(Cl)c1Cl n1(CCC)nnc2c(N(CCN(C)C)C3CC3)ncnc12.C1(C)CC1 C1(C(C(=O)N(CCCCC)C(C)C)C)CCCN(C(c2ccn(CC)n2)=O)C1 C1(NC(=O)CCn2cnnn2)CCOC(C(=O)NCC2(CO)CCCC2)C1 C(CC(=O)NCc1cn(C)cn1)(C1CC1)NC(CC=C)=O c1(CCC(CO)NC(c2ccc(F)cc2)C)ccc(Br)cc1 N1(C(Cc2c(C)ncs2)=O)CC2(CCC(NC(C3CC34CC4)=O)CC2)C1 N1(C(c2c(CC)csc2)=O)CCN(CC(C)NC(=O)C(C)CC2CC2)CC1 CC1(C)CC(NC(=O)CC2(C)CC2(Cl)Cl)CCN(C(c2nc(Cl)cs2)=O)C1 Nc1cccc(C(N2CC(CNC(C34CSCC3C4)=O)C(O)C2)=O)c1 C1(NC(=O)NCCC(CC)N2CCOCC2)CCN(C(C)C)CC1 C12(NC(COC(CC)(C)C)=O)CCN(C(=O)CCOC3CCCC3)CCC1C2 c1(C(N2C(C(=O)NCC3C(CCC)C3)C=CC2)=O)oc(SC)cc1C Cc1nn(C)c(C)c1C(=O)NCC1CCN(C(c2cc[nH]c2C2CCCC2)=O)C1 N1(C(C2(CC(C)C)CC2)=O)CCC2(CC1)C(NC(c1nccn1C)=O)CS2(=O)=O N1(C(C2(OC)CC2)=O)CCCC(NC(c2c(C)nsc2N)=O)C1 CCCCC(C(=O)N(CC(C)NC(=O)CCN(C1CCCCC1)C)C)C(C)C C1(C(N2CCC(C(CNC(C3CCCCC3F)=O)O)CC2)=O)CCC(F)(F)CC1 CCC(CC)CC(=O)N1CC2(CC)CC1(CNC(c1c(Br)nnn1C)=O)C2 c1(C(N2CCC(C#N)(CNC(C(CC)=O)=O)C2)=O)n[nH]c2c1CCCC2 C(CCCCC(=O)NC1CC(CNC(=O)Cn2ccc(C)n2)C1)OC C#Cc1ccc(C(=O)NC(C(=O)NCC(CC=C)CC(C)C)C2CCC2)c(C)c1 c1(C(N2C(CNC(C(CSC)C)=O)CC(O)C2)=O)ccc(F)c(Cl)c1 CC1(O)CCN(C(=O)CC2(C)CCCN2C(=O)C(F)=CC2CC2)CC1 c1(C(c2nnnn2C2CC(F)(F)C2)NC(c2nccs2)CC)cnc(O)s1 C1(CC=C)(NC(c2scnc2C(F)F)=O)CCN(C(C2(C)COCCO2)=O)CC1 c1(CC)cccc(C)c1NC(=O)CN(C(=O)CN1CCCC1C)CC1CC1 C1(C(N2CC(NC(C(CC)OC3CCCCC3)=O)C2)=O)CCC2(CC1)CC(=O)C2 CCC(C)(CCNC(=O)CCOCC1CC1)NC(=O)C(c1ccccc1)C c1(OCC)ccccc1C(=O)NCC1C(C)CCN1C(C1CC1CC)=O CC(C)C(O)C(=O)N1CCCCC1C1(NC(C2(Cc3nnnn3C)CC2)=O)CC1 C(CCC(O)C(=O)N1CC2(CCOC2)C1)NC(CC(C)(F)F)=O c1(CN2CC3CN(C(Cn4c(C)cc(=O)o4)=O)CC32)c[nH]c2cc(Cl)ccc12 O=C(C1=CCCN(C(=O)CCn2cncn2)C1)NC1CCn2ccnc2C1 c1(OC)ccc(C)cc1CNC(c1ccc(-n2cc(-c3cc[nH]n3)nn2)cc1)=O CC1CN(C(c2cnc3n2CCC3)=O)CC(C)N(C(c2cccc[n+]2[O-])=O)C1 N1(C(CCOC)=O)CCN(C(=O)C(C(C)(C)C)c2ccccc2)CCC1C C(=O)(C1=NOC(C)C1)N1CC(CC(CNC(C(C(C)O)NS(C)(=O)=O)=O)(C)C)C1 C1(c2ccccc2)(NC(C2C(C(=O)NCc3scc(C)n3)C2)=O)CC2(CC2)C1 Cc1ccc(CC(N2CCCC(N3CCN(C(=O)CC4(C(=O)NC)CC4)CC3)C2)=O)cn1 C1(NC(C(CCC)OC)=O)CCC2(CCCN(C(=O)C(C)(C)N(C)C)C2)C1 C1(CNC(c2[nH]cc(C)c2)=O)CN(C(=O)CC2CCC(C)(C)CO2)CCC1(F)F C(CC(C)(C)C)(C(=O)NC1CCCC1C#N)NC(C=Cc1c(C)cccc1)=O N1(CCC(=O)N(C2(CC(=O)NC(CN3CCC(C)C3)=O)CC2)C)CCN(C)CC1 C1(C(N(CCN(C(C2(CC#C)CCOCC2)=O)C)C)=O)CCC(C(C)C)NC1=O CN1CCC(=CC(N2CCC(C(F)CNC(=O)C3CC3)CC2)=O)CC1 N(C1CCCc2cccc(F)c21)C(C1C(=O)N(C)C(=O)NC1)=O CC(C)(C(=O)NN=c1[nH]c(Cl)c[nH]1)c1cccc(N)c1 CC1CC2CN(C(=O)NCCC(=O)OCCCCC(F)(F)F)CC12 N1(C(c2c(F)cc(COC)cc2F)=O)CCC2(CC1)CC2NC(=O)C1=NOCC1 c1(C(=O)NC2CC(n3cc(-c4c(C)n(C)nc4)nn3)C2)cc2c(cc1Br)OCO2 N1(C(CC(CC)CC)=O)CCc2cc(CNC(=O)CNS(=O)(=O)CC)ccc2C1 CCCCS(=O)(=O)N1CCN(Cc2nnc(-c3ccc(SC)cc3)o2)CC1 c1(C(=O)NCC2(NC(=O)CC(=O)NC3CC3)CC(OC)C2)cncn(C)c1=O N1(C(COC2(C#C)COC2)=O)C(CC(=O)NCc2ccc(O)nc2)C2CCCC12 C1(C(N(C)CCc2cnccn2)=O)CCN(C(=O)c2cncc(Cl)c2)O1 C1(NC(CC2(CN(C)C)CCC2)=O)(CF)CN(C(c2cn(C)nn2)=O)C1 c1(SC(C)C(=O)N(CC(C)O)CCNC(C2(C(C)(F)F)CC2)=O)ccccn1 C1(COC)(NC(=O)Cn2nnc(C)n2)CCCN(C(C2COC(=O)N2)=O)C1 CCC(C)CC(C)C(=O)N1CC(n2cc(-c3ncc(C)cc3C)nn2)C1 C1(C(N2CC(CNC(C3C(OCC)CCC3)=O)C(C)C2)=O)(OC)CCCCCC1 C1(C(NOCC(=O)OCC)=O)(NC(C2COCCO2)=O)CCC(C)(C)C1 Cc1cccc(C)c1C(=O)N(CC(C)CNC(=O)C(C)(C)c1ccccn1)C CN1CCN(C(C2CC(C)N2C(c2ncn(C(C)C)n2)=O)=O)C(CCO)C1 C1(OC)(CNC(=O)CC2CC(NC(C3CN(C(C)=O)C3)=O)C2(C)C)CC(C)(C)C1 N#Cc1csc(CNC(C2(NC(C3CC(F)C(=O)N3)=O)CC(F)(F)C2)=O)c1 C(=O)(CCCCCC(C)O)NCCCCNCCCNC(c1nccc(C)n1)=O c1(-c2nccc(NC(C3CCC(OC)C3)=O)c2)ccc(N(C)C)c(N(C)C)c1 c1(COCC)ccccc1-n1cc(C2CN(C(C3CC(F)(F)CS3)=O)C2)nn1 C1(C(c2ccccn2)N(C(=O)CCC2CC2(Cl)Cl)CCO)CCCCC1 CCCCC(C)C(=O)N1CCC(CNC(C2CCS(=O)(=O)C2)=O)(COC)C1 C1(CNC(=O)Cc2ccc(F)cc2)CCCCCC1NC(=O)CC1CC2CC2C1 CN1Cc2cccc(CNC(=O)C(=O)NC(c3cc(C(=O)O)no3)C)c2C1 C(=O)(C(CC(C)C)SC)N(C(C)CNC(c1cnc(O)n1C)=O)CC N(C1CCCS(=O)(=O)c2ccccc21)C(=O)NC1(c2cccc(Br)c2)CCCO1 C(=O)(CC1=CCN(C(=O)C(C)(C)C(C)C)CC1)NCc1c(C)nc(F)cc1 C1(C)(COC)CC(NC(=O)CNC(=O)C2CC2)CN1C(c1cccc(CO)c1)=O CC(C)S(=O)(=O)CC(=O)NC1CCCCC1CNC(C1CCCC12OCCO2)=O CCCCC(C)C(=O)NC(C(=O)NC1CCCCC1(C)O)C1CCC1 CCCCC(=O)C(=O)NC1C2CCC1N(C(=O)CC13CCCN1CCC3)C2 Cc1oc2ccccc2c1-c1nc(CCO)nn1-c1ncnn1C N1(c2n(CC(=C)C)c(C(c3ccc(F)cc3)C)nn2)CCCC2CN(C)CC12 CCC(C)(C)CN=c1nc2c(ncn2C)c(NC2CCCC3(CC2)CC3)[nH]1 S(=O)(=O)(c1cccc(C)c1C)NCC1(C)CCCN(C(C=CCCC)=O)C1 c1(CN2C(C(=O)Nc3cc(Cl)ccn3)CC3CC32)cn2ccccc2n1 C(=O)(CCCCCCN=[N+]=[N-])N1CCC(N(C)C(c2cc(=O)n3nccc3[nH]2)=O)C1 n1(CC)nc(C(=O)N(C)CC2CCN(C(C3CC4CC3C4)=O)C2)cc1C N1(C(C2C(C(=O)OC)C2)=O)CC(CNC(=O)C(F)(F)CC2CC2)CC1(C)C C1(C(N2CC(CC)C2)=O)CCC2CCC1N2C(=O)CS(C)(=O)=O c1(C(N2CC(C)C(NC(c3c[nH]nc3F)=O)C2)=O)ccc(Br)cc1N(C)C C1(C(=O)NCCCSCCO)(SC)CN(C(=O)CCCF)C1 N12CC3CCCC3(C1)C2.c1(NCc2ccnc(N(C)C)n2)ncc(C#N)cc1F Cc1[nH]c(C)c(C(=O)N(C(C)CNC(=O)C(c2ccc(Cl)nc2)(C)C)C)c1C CCC(CN(C)C)C(=O)NC1(C2CCCCN2C(=O)Cc2c[nH]nc2O)CC1 C1(NC(C2C(OC)(OC)CC2)=O)CCC(NC(=O)CSc2nccn2C)CC1 C1(COC)CCc2sc(C(=O)NCCCCc3cnc[nH]3)cc2C1 C(C(C)(C)C(C)(C)C)NC(CNC(CNC(C(C)C1CCCC1)=O)=O)=O N1(C(c2cnc(OC)nc2)=O)CCC(CNC(c2cnco2)=O)C(C)C1 C12(CSC)CCOC1CN(C(=O)OC(C)(C)C)C2.C12CCC(C1)NC2=O Cc1ccc(O)cc1C(=O)NCCOC(C)(C)CNC(C1CC2CCCC2C1)=O NC1CC(NC(c2ccc(-c3cnco3)nc2)=O)c2ncccc21 C(CC(CNC(C)=O)NC(=O)COc1ccccn1)OC C(=O)(C1=NN(CCO)C(=O)CC1)NC1C(C)CN(C(C2(n3cnnn3)CC2)=O)CC1 C1(n2cc(-c3ccc(C(=O)O)o3)nn2)(OCC2CCOC2)CC2(CCCCCC2)C1 c1(CNC2CCC(C(=O)NCC(O)CO)C2)cc(Cl)nc(Cl)c1 N1(C(C2CCSC2)=O)CC(C2CC2)(C(N2CCC2C2CCC2)=O)C1 C(CC(C)C)(C(=O)N1CCN(C(N)=O)C(C)C1)NC(COc1cccc(C)c1)=O Cc1cc(C=CC(N2CCC(CCNC(=O)CCC3CCCO3)C2)=O)c[nH]c1=N C(=O)(C1=CCCCC1)N1C(C)C(C(=O)NCCCS(N)(=O)=O)CC1 C(N=c1cc(C)[nH]c(=NCC2CCCC2C)[nH]1)c1ncc(CC)o1 Cc1ccc(CCNC(c2ccc(Cl)o2)c2nnnn2C2CC2)cc1[N+](=O)[O-] N1(C(C2CCCS2)=O)CCN(C(c2cc3ccncc3s2)=O)C2CCCC12 N1(C(C(CC=C)NC(=O)OC(C)(C)C)=O)Cc2nncn2CC1C(=O)OC c1(NCC(=O)NC2C(NC(CCC=C)=O)CC2)cccc(C#N)c1 N1(C(C(C)NC(C)=O)=O)CC(NC(=O)C(C)(C)n2cncn2)CC12CCCCC2 C1(C(=O)NC2CC(NC(C34CCN(CC3)C4)=O)C2)CC2CC1C1CC21 c1(-c2ccc(C(N3CC4CCCC3CC4)=O)c(F)c2)cc(F)c(CS)c(F)c1.CN Cc1ccccc1C(=O)NCC(=O)NCC12CC1CN(C(C1(O)CCSC1)=O)C2 C1(CNC(=O)NC23CC(Cc4ccccc4)(C2)C3)CCC2(CC1)CNC(=O)C2 c1(NCC(C)C)cccc(C(N2CC3CC3(CNC(C3(O)CCC3)=O)C2)=O)c1 N1(C(C(C)(C2CC2)OC)=O)CCC(C2CC2)(NC(c2ccc(S(N)(=O)=O)s2)=O)C1 N1(C(CCC2(C)N=N2)=O)CC(OCc2ccccc2)C2(CC2)C1 C12(CNC(C3C(CC)CCO3)=O)CN(C(C3CC(=O)NC(C)C3)=O)CC(F)(C1)C2 c1(CC)ccc(C(=O)NC2CC(NC(C3(C)CCC3)=O)C2)cc1[N+](=O)[O-] c1(CC=C)cncc(C(=O)N(C2CC(F)(F)C2)CCC)c1 c1(OC)cccc(Cl)c1C(=O)NC1CC1CNC(c1ccc(CN(C)C)[nH]1)=O C(C)(CS(=O)(=O)N(C)C)NCC1(CC(=O)NC(C)C)CCOCC1 C(=O)(CCS(N)(=O)=O)NCC(CCCC)NC(C1CCC1CF)=O N(C1CCc2c(Br)cccc21)C(C1(C)CCN1C(=O)CCN1C(=O)C=CC1=O)=O C1(CC)CCN(C(=O)Cn2ncccc2=O)C1CNC(C1CC(F)(F)C1)=O c1(-c2ccc(C(=O)NCCC(C)(C)NC)s2)ccc(C(=O)NC2(CF)CC2)cc1 CCCCC(O)CC(=O)N(C)CNC1CC(F)CN1C(c1cnc(C(N)=O)cn1)=O c1(CCC(=O)NCC2CCCN(C(C3(OC)CCC3)=O)C2)cccc(Br)c1F C(=O)(CCN1CCCC1)N(CC(=O)N(C)SC1CC1)CC.C1(NC)(C)CC1.CCCOC C1(CC)CC2CCC(C1)N2C(=O)NCC1CCCC1c1ccccc1 C(CC(C)C)(C(=O)N(C(C)CN(C(=O)CSCc1ccsc1)C)C)OC CN1CCC2CCN(C(c3ccc(O)cc3Br)=O)C2C1 CC1=NNC(=O)C1CC(=O)NCC(C(C)C)NC(C1CCS(=O)CC1)=O c1(C(N(CCOCCNC(CC(C=C)C)=O)C)=O)cn2nc(C)cc2[nH]c1=O c1(N(C)CC2CCCN2C(=O)C(O)C2CC2)cc(OCCO)ccc1[N+](=O)[O-] C(=O)(C(F)(F)CO)N(C1CN(C(=O)C=C2CCC(C)C2)CC1O)C CC(C)(C)C(O)C(=O)NCC1CN(C(c2cccc(C(F)(F)F)c2C)=O)CCO1 c1(C(=O)NCCCC(=O)NC2CN(C(C)=O)C2)cnnc(O)c1 c1(OC)cc(C)c(C(N2CCCC(NC(=O)CNC(C)=O)C2)=O)cc1OC Cc1cc2c(cc1Br)CN(C(=O)NNc1nccn1C)CC2 c1(C(N2CC(NC(C(CC)n3cncn3)=O)C(C)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(O)C(=O)N1CCC(n2cccn2)(CNCc2cccc(F)c2)CC1 c1(COC(C(c2cccc(C#N)c2)O)=O)c(F)c(F)c(F)c(F)c1F N1(C(C(CCC)C)=O)CCC(CO)C(NC(=O)Cc2ccc(Cl)cn2)C1 C#CCC(CC(=O)NCCOc1ccccc1)NC(C1(C#C)CCCC1)=O C1(C(=O)NCC(C)NC(c2c[nH]c3nccc-3c2)=O)CCOCC12CCCCC2 C1(CNC(COCC)=O)CCCC2(CN(C(C34CC(CC(F)F)(C3)C4)=O)C2)O1 c1(CC)ccc(C)cc1NC(=O)C(C(C)C)NC(C1(C#N)CCCOC1)=O C12(C(=O)NCC3C(C(=O)NC(c4cnc(C)s4)C)CCO3)CCC(CC1F)C2 N1(C(COCC(=C)C)=O)CC2(CCN(C(=O)C(C)c3ccsn3)C2)C1 C(C)(C)(C(C)CC(=O)NC(c1ncccn1)C)NC(C(C)n1cccn1)=O c1(C(=O)NC(CC=C)CNC(=O)C(C)C2CCCC2)cc2occc2s1 C1(N(C(CC=C=C)=O)CC)CCCN(C(c2ccn(C)c2-c2ccccc2)=O)C1 N1(C(C2(COC)CCC2)=O)CC2CC(C(=O)N(C3CCCC(C)(C)C3)C)(C2)C1 N1(C(=O)NCC2CCN(C(=O)OC(C)(C)C)C2)CCOC(C2CC2)CC1 N1(C(CC2(NC(C3C(C)C3)=O)CCC2)=O)CCC(N2CCCC2)C1 CC(C(=O)NCCOCC(=O)NCC1(Cl)CC1(F)F)C(C)(C)C c1(NC(N(CCN(c2nc(SC)nc(C(F)(F)F)c2)C)C)=O)cc2cnccc2[nH]1 C1(C(=O)NCCc2cnc(-c3ccccc3)[nH]2)CCN(Cc2nccs2)CC1 CCC(C)(C(=O)NCC1(F)CCC(CNC(=O)C(=O)NC2CC2)CC1)C(N)=O C(=O)(C1=CCCN(C(c2ccc3occc3c2)=O)C1)NCc1ccc(C)nc1 N1(C(C(C(=O)N(C)C)(C)C)=O)CCC2(NC(=O)Cn3cccnc3=O)CCCC12 O=C(C#CC1(C(F)(F)F)CC1)NC1CCC1NC(c1ccn(C(F)F)n1)=O N1(C(c2c(CC)ncs2)=O)CC2CN(c3cc(C#N)ncn3)CC12 c1(C(c2n(CC)nnn2)NCC2(C)CCOC2)cn(C)nc1-c1ccccn1 c1(NC2CCN(C(C(c3cccc(F)c3)C)=O)C2)ncnc2sc(C(F)F)nc12 CC1CCCCN1C(=O)CN1CCCC(CCNC(=O)CC(C)(C)C2CC2)C1 C1(N(C(=O)CCNC2C=CCC2)C(COC)C)CC2(CCNCC2)C1 C1(COC)(CNC(C2(C)CCOCC2)=O)CCCN1C(=O)C(c1cccnc1)O C1(CC(=O)NCC2C3CN(C(c4c(C)noc4)=O)C2C3)CN2CCC1CC2 Cc1cc(C(N2CCC(NC(=O)COCC(F)F)C(CO)CC2)=O)cc(N)c1Cl N1(CC(N2CCC(NC(c3n(C)nc(O)c3)=O)C2)=O)CCCC2(CC2)S1(=O)=O c1(C(=O)NCCCC(C)NC(c2nnn(CC)c2C)=O)cc(C)c(C(F)F)cn1 C(=O)(C1CCCc2cc(C#N)ccc21)NCCCN(C(=O)COCCOC)CC Cc1cccc(NC(=O)NCCCCOc2ccc(Br)cc2)c1F C1(C(=O)NC2CN(CC)C2)CCCCN1C(c1csc(=N)[nH]1)=O CC(CC(N)=O)C(=O)NC1CCCN(C(c2cc3n(c2)CCC3)=O)C1 C1(CCO)(OC)CCCCC1.c1(C(CCC2CCCO2)N)nnnn1CCC1(C)CC1 CC1CN(C(=O)Cc2cccc(F)c2O)CCCN1C(C1CC(=O)NC1(C)C)=O C1(CC(N2CCN(C3CN(C(c4ccc(Cl)s4)=O)C3)CC2)=O)NC(=O)NC1=O C1(O)(C(=O)NCC(C2CCCC2)NC(CC(CC)C)=O)CCCC(C)(C)C1 c1(C(=O)NC2(CCNC(c3c(C)[nH]cc3)=O)CC2)csc2c(F)cc(F)cc12 C=CC1CN(C(C2(O)CCSCC2)=O)CC1NC(c1ccc(OC)cc1C)=O N1(CC(=O)N(C(C)CNC(C2CC(C3CC3)C2)=O)C)C(=O)NC(C)(C)C1=O O=C(CCCCC(F)F)NCCC1CC(F)(F)CN1C(c1ccc(F)c(Cl)c1)=O Cc1cnn2c1CN(C(C1COCCN(c3nccnc3C(N)=O)C1)=O)CC2 c1(SC)ncc(N)c(C(=O)NC(CO)C(C)NC(c2csc3cncn23)=O)n1 C1(N(C(COCC#C)=O)C)CN(C(c2ccc(-c3cccc(Cl)c3)s2)=O)CC1O C(C)(CCCN=c1[nH]cc2ncnc-2[nH]1)NC(CCCc1ccc(OC)cc1)=O CCCCC(F)C(=O)N(CC(=O)NC1CN(C)CC1(F)F)CC c1(CC(=O)N(C2CCN(C(C=C(CCC)C)=O)C2)C)ccc2c[nH]nc2c1 C1(C(=O)NC(CC)CO)C2CC1N(C(=O)CN1CCC(C)CC1)C2 N1(C(C(C)(F)c2ccon2)=O)CCCC2(C1)CN(C(C1CCC(C3CC3)C1)=O)C2 C#CCCCC(C)C(=O)NCC(C1CC1)NC(c1cc(F)c(F)c(F)c1)=O N1(c2nnc(CC)o2)CCC(C2(NC(=O)C3=CS(=O)CCC3)CC2)CC1 CC(CC1CC1)C(=O)NCCCOCCNC(=O)C(C)(C)c1nncn1C c1(C(=O)NC(c2nnc(Br)n2C)C)ncn2c1CCCCC2 N1(C(c2c(CNC(C3CCS3(=O)=O)=O)occ2)=O)CC2CC1CO2 N1(C(CCN(C(=O)CN2CCC(F)CC2)C)=O)CCOCC1c1nc[nH]n1 Cc1ccc(C(C)NC(C2CC(NC(c3cn(C(C)C)cn3)=O)CCO2)=O)nc1 N1(C(COCCOC)=O)CC2(C(N3CCC4(C3)CN(C)C4)=O)CC1CCO2 CC1(O)CCCC1NC(=O)CC1CCCN1C(=O)CN1C(=O)CNC1=O N1(C(CCOCCCNC(C(CC)=CC)=O)=O)CCCC1(C)C(C)(C)C c1(N(C(C)=O)C)ccc(Cl)c(C(N2CCC(CNC(C34CCC3C4)=O)CC2)=O)c1 CC1CCCC(C)N1CCC(N1CCN(C)C(CNC(=O)C(C)CN(C)C)C1)=O C1(CC(=O)NC(CCC(=O)NC(C(=O)OC)c2ccco2)C)C(C)(C)C1(C)C C(CCC(CCC)NC(c1sccc1CC#N)=O)NC(CCSCCC)=O CCC(CC(=O)c1ccncc1)C1CCC1.C1(CCN)(CNC(C2(N)CC2)=O)CC1 c1(CC)[nH]nc2ccc(C(=O)NC3CC(NC(C4CCC4COC)=O)C3)cc12 C1CN=C2NC(=CS2)C(=O)N2CCC1C2.n1(CC(=O)OC(C)(C)C)cccn1 C(C(O)CC(=O)NC1CN(c2ncco2)C1)NC(C1(C)CCC1)=O c1(C(=O)NCC2CN(C(C(CCC)=CCC)=O)C(C)C2)ccc([N+](=O)[O-])[nH]1 N1(C(c2cc(OCC)ncc2)=O)CCCC2C1CCCN2C(=O)Cn1cccn1 C12(CNC(CC=CCC)=O)CCC1CN(C(=O)CCc1ncc(C)[nH]1)C2 C1(C(N2CCC(NC(C(C)(C)SC)=O)C2C(C)C)=O)CCC2(CCC2)O1 C1(CCC(=O)NCc2ccc(F)cc2)CCN(CC(F)CO)CC1 CCCCC(C(=O)NCC(C)C(=O)NC)NC(c1cncc(C#N)c1)=O c1(C(N(C2CCN(C(C3(C)CC(C)C3)=O)C2)C)=O)ccccc1S(=O)(=O)C(C)C C12CC3(C1)CC(C3)C(=O)N2.c1(C(=O)NCCC2ON=C(C)C2)ccc(F)cc1 C=CC1CCCN1CC(C1CC(OC)C1)OCC Cc1ccc(CNC(C2(CNC(=O)C(CO)OC)CC23CCC3)=O)c(O)c1 c1(CCC(=O)NC(CN(C(c2cncc(C)n2)=O)CC)C)cccc(F)c1F C(CCC)(C(O)C(=O)N(C)Cc1cn(CC)nn1)NC(C(C=C)(F)F)=O C(CCC(=O)NCCC1(C(=O)NC(C)(C)CCF)CCC1)OCC CCCCCC(C)(C)C(=O)NCC(C)(O)CNC(C1CC1(C)C)=O C(=O)(C(CC(=C)C)OC)NC1(C(=O)Nc2cn(CCC)nc2)CC(CO)C1 c1(C(N(C(CNC(C(CC=C)CC)=O)C)C)=O)ccc2c(c1)nc(O)n2C N1(c2c(C(C)=O)cccn2)C2CCC1CN(C(C1CC1C1CC1C)=O)CC2 c1(C(=O)NCC(CC)NC(C(COCC)C)=O)cc(SC)nn1C N1(C(CN2CC(C)C2)=O)CCC(CNC(=O)CN2CCNC(=O)C2)C(C)C1 N1(c2cc(C)nc(N3CCC(CC4CC4)C3)n2)CCCC2(CCCCO2)CC1 n1(CC)cnc2c(N(C)CCC3CCOCC3)nc(N3CC4CCC4(C)C3)nc12 c1(C(=O)NCC#CCNC(C(CC=CC)C)=O)c(C)[nH]c2ncccc12 c1(C(=O)NC23CC(CNC(C(COC)C)=O)(C2)C3)ccnnc1O N1(C(COCCC#C)=O)CC2CCN(C(c3cc4nc(C)sc4[nH]3)=O)C2C1 c1(CN(C)C(c2ccc(Cl)s2)=O)ccc(CNC(=O)C(c2cccnc2)O)cc1 N1(C(CCC=C)=O)CC(CNC(c2cccc(F)c2C(C)C)=O)C(F)(F)C1 c1(NC(N(C2CC2)CC)=O)nnc(C(C)C)o1 C1(CNC(c2ccnc3[nH]ncc23)=O)CN(C(C23CC(C2)C3)=O)CCC1(F)F C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(C)CN(C)C)CC2CCCC12 c1(C(=O)OC)ncn2c1CN(C(=O)N(C)C(c1ccc(C(C)C)cc1)C)CC2 N1(C(c2ccc(NC)cc2)=O)CCC2C(C(=O)N(C(C)C)CC3CCOC3)C2C1 CCC1=NOC(C(=O)N(C2(C(=O)NCC(C)O)CC2)C)C1 C(=O)(CC(O)CC(C)C)N1C(CNC(=O)CC2(CO)CC2)CC(OC)C1 CCCCC(CNC(=O)C=CSC)NC(=O)Cc1ccnn1C1CCC1 c1(C(=O)NC(CC)(C)CNC(C2CCNC2=O)=O)cc(OC(C)C)ccc1N CC(C)C(C)(O)C(=O)N1CC(O)(CCNC(c2c[nH]cc(F)c2=O)=O)C1 Cc1cc(C(=O)NC2CCCCC2NC(C2COC(=O)O2)=O)c2ccccc2n1 c1(NC(=O)CN2CC3C=CC2C3)nc2c(s1)CC(NC(c1ccccc1)=O)CC2 C1(O)(C(C)C)CCCN(C(=O)C=CC2CCN(C(=O)C(=O)NC(C)C)CC2)C1 C1(CCO)(N(C(C(OCC)OCC)=O)C2CC2)CN(C(C2SCCC2C)=O)C1 c1(C(N(CCCN(C)C)CCNC(C2CC2(C)C)=O)=O)cn2cccc(F)c2n1 CCCCC(O)C(C)C(=O)N1CCC(C(N2CC(c3cc(O)no3)C2)=O)C1 S(=O)(=O)(c1ccc(NCCC(C(C)C)SC)c(C#N)c1)N1CCC(OCC=C)C1 c1(C(=O)OC)cc(C(=O)NC23CC(CNC(=O)C(C)N(C)C)(C2)C3)cn1C c1(N2CCCC(C)(NC(=O)CCc3ccc(Cl)s3)C2)ncc2scc(Br)c2n1 CC(C(C(=O)NCC1(C)CC1)N1CCCC1Cc1ccccc1)c1ccccc1 Fc1cc(Br)cc(-c2noc(C34CCCCC3C4Br)n2)c1F C1(CNC(=O)CCOCC(F)F)CCN(C(=O)CN2CCC(=O)CC2)CC1(F)F Cc1ccc(C(=O)NC2CCCC2(C)CNC(c2nsnc2O)=O)cc1C C1(NC(C(C)(O)C2CC2)=O)CC(F)CN(C(c2sccc2-n2cccc2)=O)C1 C(=O)(CCCC(F)(F)F)NC(CCOC)C(N1CCC(=C(F)F)CC1)=O C12(CCOCC1)C(=O)NC2.C1(NC(C(C)SC)=O)CCN(c2ncc(I)cn2)CC1 CCCS(=O)(=O)C(C)C(=O)N1CCOC(CNC(C2(C#N)CCSCC2)=O)C1 N1(C(c2c[nH]nn2)=O)C2CCC1CC(n1cc(-c3ccns3)nn1)C2 Cn1cc2cccc(C(=O)NC3CC3CNC(c3cccc(N)n3)=O)c2n1 CC1CCC=C1C(=O)N1CCN(C(c2cc(=O)c(Br)c[nH]2)=O)C(CO)C1 c1(-n2cc(-c3ccc(C(=O)OC)o3)nn2)ccc(C)cc1C C(N=c1nc2c(cnn2C)c(NC2CCSC2)[nH]1)C1C(CC)CCOC1 C(=O)(CCCS(C)(=O)=O)N1CC(CNC(c2cc(C#N)oc2)=O)C(CO)CC1 CS(=O)(=O)c1ccccc1CC(N1CC(CCNC(C2(F)CCCOC2)=O)C1)=O C1(NC(C(C)OCC=C)=O)CCCN(C(=O)Cn2cc(CC)cn2)C1 c1(CNC(c2c(C)nsc2)=O)ccc(C(=O)NC2CC2)cn1 C1(CC)CN(Cc2nc(C3OCCO3)cs2)CC(C)S1(=O)=O c12cnc(nc1O)Cc1nn(-c3c(CC)cccc3)c-2n1.CC(C)C.C(C)(OC)OC CC1=C(C(=O)NC2CCN(C(c3ccn(C4CC4)n3)=O)C2)C(C)(C)CCC1 C=C(C)C1OCCCC1C(=O)NCCCCN(C)C(C1CCCCC1CC)=O C1(C(=O)NC2(C3CC3)CCN(C(CCOCC)=O)C2)CN2CCN1CC2C C(=O)(C1CCSc2ccccc21)N(CC(C)NC(C1CCN(CC)CC1)=O)C N1(C(CCC(=O)N(C)C)=O)CCC(O)CC1C(=O)NOCCC(C)O C#Cc1nccnc1NC(C1CC12CN(C(=O)Nc1ccccc1Cl)C2)=O N1(C(c2ccc(Cl)c(F)c2)=O)CC(N=c2ccnc(CO)[nH]2)C1 c1(C(C(=O)NCC2CCN(C(CC(C)F)=O)C2)O)cccc(Cl)c1 N1(C(CC2(N(C)C)COC2)=O)CCCC(CCNC(=O)C(O)C(C)C)C1 C1(NC(CC(C)SC)=O)CCC(n2cc(C3CC3COC(C)(C)C)nn2)CC1 N1(C(CNC2C(NC(=O)OCC)C2)=O)CCCC2(CCCO2)CC1 CN1CC2CC1CN2C(C1COCCN1C(C1CCC2(CCC2)O1)=O)=O C1(C)(CNC(CCC=C(C)C)=O)CCCN1C(c1ccon1)=O N#Cc1c(N2CCCC(C(=O)Nc3cnsc3)CC2)cccc1F c1(CC)cccc(CCCn2nnnc2C(c2ccc(CSC)s2)OC)c1 C(=O)(C(CCOC)OC)NC1(CCC(=O)NC(c2n(CC)ncc2)C)CCC1 C1(NC(C2C(C)CCN2C(=O)Cn2cc(C#N)cn2)=O)CCC(C2CC2)C1 C(C1=CCCCC1)NC(C1C(CNC(C2(CCC)CC2)=O)OCC1)=O c1(CC)[nH]ccc1C(=O)NCCCC1CCCN1C(C1CSCCS1)=O CCC(C#N)C(=O)N1CCC(N2CCN(C(=O)Cc3csc(S)n3)CC2)C1 N1(c2ccnc(OC)n2)CCC(NC(=O)C(N2CCOCC2)C)C(F)C1 c1(C(N2CCCC(C(=O)NCCCC(F)(F)F)(CO)C2)=O)c[nH]nc1[N+](=O)[O-] Fc1ccc(N2CCOCC2CCNCC2COC(C3CC3)C2)cc1 c1(C(=O)NC(CC(C)NC(c2ccc(C)c(Cl)c2)=O)C)c(F)ccc2c1OCO2 C1(C(=O)NCCC2C(C)=NNC2=O)CC2(CC(NC(C3(CCF)CCC3)=O)C2)C1 C12(C(=O)NCCCC3OCCN(C(C4CC=C(C)CC4)=O)C3)CCN(CC1)CC2 C1(CNC(C=CC)=O)CN(C(C2CCC2(OC)OC)=O)CC12CC2 C=CCC(C)(C)CC(=O)NC1CC(CNC(c2ccc(CC)s2)=O)C(O)C1 C1(NC(c2c(CC)noc2C)=O)CN(C(=O)C=Cc2cncn2C)CCC1C C(=O)(C(F)(F)C(F)(F)Cl)NC1CCC(CNC(c2c(C)snc2)=O)CC1 C(CCC(C(=O)NC1CCCC1(C)O)NC(=O)C(COc1ccccc1)OC)OC N1(C(c2c(C)ocn2)=O)CC(NC(c2ccc(Cl)s2)=O)C(C2CC2)C1 C1(C)(C(=O)NC2CC(CCNC(CN(S(C)(=O)=O)C)=O)C2)CCCC1 Cc1cc(C(=O)OC2CC2C2CCCC2)c2cnn(-c3ccccc3)c2n1 n1(C(c2cccs2)C)nc(-c2ccccc2)nc1-c1cc(Cl)ns1 c1(C(=O)NC2CN(C(=O)CCC3CCCC3)C2)c(Cl)cccc1Br CC(C)C(C)(CNC(=O)CCOC1CC1)NC(c1ccc(CO)cn1)=O CC(C)(C)CC(O)C(=O)NC(C)(C)CC(F)C(=O)N1CCCC(C)(CO)C1 C1(CC(=O)NCCN(C(=O)CCc2ccc(C)s2)CC)COCCN1CC C1(CC(=O)OC(C2CN(C(C)=O)C2)=O)CCCNC1C.c1(C2CCC2)nn[nH]n1 C1(NC(c2scc(C)c2)=O)CCN(C(c2ccc(C(O)CF)cc2)=O)C1(C)C N1(C(CNC(CC)=O)=O)C2CCC1C(NC(=O)C(F)n1ccnc1)C2 N1(C(C2CCN(C(=O)CCc3cncnc3)C2)=O)CC2CCC(CC2)C1 C1(OC(C)C)CCCN(C(=O)CCCNC(=O)CC2C=NN(C)C2=O)C1 C1(CNC(=O)CCc2cnoc2)CCCC(NC(=O)CC2CCOCC2)C1 c1(C(=O)NCC2CCN(C(C(C)O)=O)CC2)cc2c(Br)cc(Cl)cc2[nH]1 N1(C(C(C(C)C)OC)=O)CCC2N(CC=CCl)CCCCC2C1 CCC1(CC)CN(C(C)=O)c2ccccc21.C12CC(C1)NC(=O)C2 Cc1ccc(CNC(C2CN(C(=O)CC3CCCC3(F)F)C(C)(C)C2)=O)cc1C CC1CN(C(c2ccn(C3CCCC3)n2)=O)CCC1NC(c1csc(Cl)n1)=O C12(NC(C(=O)NC3CC3)=O)CCC(CC1n1cc(CN3CCSCC3)nn1)C2 C(=O)(CCC(=O)NN(C)C)N(CCO)C(c1cccc(F)c1)C.CC(C)CO c1(NC(=O)NC2CCCCC2)ccc(-c2csc(N3CCC(O)CC3)n2)cc1 N1(C(c2c(CC)nccn2)=O)CCC(CNC(C2CCCSC2)=O)C12CCC2 C(=O)(C(C(C)(C)C)OC)NCCC(C)(C)NC(C(CC)CC1CCCCC1)=O c1(CC(=O)NC2CC(F)(CNC(C(CC)=CC)=O)C2)sc(C2CCC2)nc1C O=C1CCC(CCC(=O)NCCC2(CNC(=O)CN(C3CCC3)C)CC2)CN1 c1(C(c2nnnn2CCCF)NCC(C)C(F)F)cc(C(=O)N(C)C)cc(Br)c1 CC(CCN=c1ccnc(NC2CCOCC2)[nH]1)C(F)F.C1CN(C)CCO1 CCC(C)(CNC(c1cc(-c2csc(C)n2)c[nH]1)=O)NC(=O)CCc1ccsc1 N(C1CCCc2ccccc21)C(C1(F)CN(C(c2c(C)ccnn2)=O)C1)=O C(=O)(CS(=O)(=O)Cc1cnn(C)c1)N(CC(C)CNC(=O)C=CBr)C C#CC1CC2CCC1N(C(C1CCCN1C(=O)C=CC(C)(C)SCC)=O)C2 N1(C(CN2CCCC(N(C)C)C2)=O)CCC(NC(C2(O)CCCC2)=O)C(O)C1 C#CCCCCC(=O)NC1CCCC1CNC(=O)CC(C)SC CC1C(NC(c2c[nH]cc(Cl)c2=O)=O)CCN1C(=O)CCN1CCCS1(=O)=O c1(CCC)sc(C(=O)N(CCCNC(=O)CC(C)F)C2CC2)cc1Br C1(C(N(C(C)(C)CC(N2CCC(C)(CO)C2)=O)C)=O)CCCC2(CC2)C1 c1(NC(CC)=O)ccc(NC(c2cc(CC)n(CCO)n2)=O)cc1C CC1(C)CN(C(=O)C2=NOC(C)(C)C2)C(CNC(c2ccc(Cl)cn2)=O)CO1 CC(C)(C#N)CC(=O)N1CC(O)(CCNC(=O)C(c2cc(F)cc(Cl)c2)=O)C1 C(=O)(C1=CC2(CCN(C(C3CC4(CC4)C3)=O)C2)C1)NCCCCC#C Cc1ncc(N)cc1C(=O)NCC1CCCCN1C(=O)C1=CCCC1C C1(C(=O)NCCN(C(CC2CCN(C)C2)=O)C2CC2)CCCNS1(=O)=O S(=O)(=O)(c1ccc(NCC2CSCCS2)c(C#N)c1)N1CCc2c(nc(C)s2)C1 CCCC(C(=O)NC1CC(F)(F)CC1C(=O)Nc1ccc(OCC)cc1)C(C)C C(=O)(C(O)CC(F)F)N1CC(O)(C(C)(C)NC(C2CC2[N+](=O)[O-])=O)C1 N1(C(C23CC(NC(C(COC)OC)=O)(C2)C3)=O)CCC(CO)C(O)C1 N1(C(C(C)Oc2ccc(COC)cc2)=O)CC2(CCN2C(C2CC2(F)F)=O)C1 Cc1ccnc(C)c1C(=O)NCCC(O)CNC(c1cn(C)c(=O)n1C)=O C1(NC(CSCC#C)=O)CC(CC(=O)NCCCC)C1 c1(C(=O)NC2CN(C(CCCC)=O)CC2c2ccc(F)cc2)cc(Cl)cnc1O N1(CCCCNC(CNC(C)=O)=O)CCCN(C(C23CCCC2C3(F)F)=O)CC1 C#CC1(NC(c2ccnc(CNC(C3CC3Cl)=O)c2)=O)CCC(C)(C)C1 C1(NC(c2cc(OC)n[nH]2)=O)C2CCC(C2)C1C(N1CCCCC1CO)=O C=CC(C)CC(=O)N1CCC1C(=O)NC(C)C(C)SC Cc1ccc(CCNC(c2ccc(-c3cn[nH]c3)cn2)=O)cc1 c1(CC(=O)NC2CCC2c2cccc(-c3nn[nH]n3)c2)cccc(F)c1F Cc1cnccc1CN(C(C1CCCCC1)C(=O)NC1CC1)C C1(CNC(CNC(c2c(C)occ2)=O)=O)CCC(C)N(C(=O)CC2CC(CF)C2)C1 C1(C(=O)NCC(=O)NC(C)C2CC2)CCC12CN(C(C1CCCO1)=O)C2 CC(C)CC(C(=O)N1CC(CCNC(=O)C(C)N(C)C)C1)c1ccccc1 C1(C(N(C)CC2CN(C(c3[nH]ncc3C#N)=O)CCO2)=O)CS(=O)(=O)CC12CC2 c1(C(=O)NCC2(NC(C(C)SC)=O)CCCCC2)ccnc2c1ncn2C c1(CNCC2(COC)CC=CC2)cc(N2CCCS2(=O)=O)ccc1F CC(CS(=O)(=O)N1CC2C3CCC(C3)C2C1)C(F)(F)F N1(C(C2CC(OC)C2)=O)CC(NC(=O)COc2cc(C)ccc2F)CC1(C)C Nc1c(C(=O)NC2CC(CCNC(=O)C(F)n3cccn3)C2)ccc(Cl)c1F c1(C(=O)NC(CC(C)NC(c2c(OC)n[nH]c2)=O)C)ncc(Br)cc1OC c1(C(N2CCCC(CNC(C(CC)(F)F)=O)(CO)C2)=O)[nH]cc([N+](=O)[O-])c1Cl c1(N(C(C(=O)Nc2c(C)cccc2C)C)C)cc(F)c(Cl)cc1Cl N1(C(c2ccc(C)cc2Br)=O)CCCC2CN(C(=O)C(O)C(F)F)CCC12 N1(C(CN(C(C2C(C)OC(=O)N2)=O)C)=O)CCC2(C1)CN(C)C2 CCC(CC)CCCC(=O)N1CCN(C(=O)CCCNC(C)=O)C(C2CCC2)C1 C12CN(CCS1(=O)=O)C(=O)C(=O)NCC2.C1(CC=O)CC2(CC2)CO1.C1(N)CC1 c1(C(=O)OC)cncc(-c2csc(NC(=O)C(C)CBr)n2)c1 CCCC(C)(C)C(=O)NCC1CC1NC(=O)COCc1ccc(C)cc1 c1(CC)ccc(F)c(C(N2CCC(NC(C3(F)CC=CC3)=O)C(O)C2)=O)c1 N1(C(CCC)=O)CCCC(C(=O)NCC(C)CNC(c2ccc(C)cc2)=O)C1 C(C(=O)NOCC1(C)CC1)(NC(C(COC)OC)=O)SC N1(C(C(C=C)(C)O)=O)C2CCC1(CNC(c1scnc1COC)=O)CC2 C1(C(=O)NC2C(c3cn(C)nc3)C2)CN(C(=O)CC(C)(C)C)CCO1 CCC(CCCC(=O)N(C1CCCCC1)CC1CC1)NC(=O)C(C)N(C)CC CC(CC(=O)NC1(CC(=O)NCCC2OCCC2(C)C)CCC1)C(F)(F)F c1(C(C)NC(C(F)=CC)=O)ccc(CNC(c2cnn(C3CCC3)c2C)=O)cc1 C1(C(=O)NCC#CC(=O)Nc2cncc(OCF)c2)CN2CCN1CC2 c1(C(N2CC(OCc3c(OC)cc(F)cc3)C2)=O)cc(Br)cc2[nH]ccc12 c12ccc3c(c1)CN(CC3)C(=O)CNC2=O.C(CCCCO)N(C)C1CC1 C1(C(=O)NCC2(O)CCN(C(C3CCS(=O)CC3)=O)C2)CCC2(CCC2)CO1 n1(CC(=O)NCC=CCNC(c2c(C)n(CCO)cc2)=O)c([N+](=O)[O-])cnc1C c1(C(N2CC(OCC(=O)NCCOC3(F)CC3)C2)=O)cncc2c1CCNC2=O C(N=c1nc(N2CCC(C)(CO)C2)c2c([nH]1)CSC2)C1N(C)CCC1 N1(C(Cc2cc(COC)on2)=O)CCC(NC(=O)C(C)OC2CCC2)C(O)C1 C1(CCNC(C(C)NC(COC)=O)=O)CCCCN1C(C1(c2nc[nH]n2)CC1)=O c1(NC(C(CCSCC)NC(C2CS(=O)C2)=O)=O)cc(CC)cc(O)c1 C(CCC(O)C(=O)NCC#CC(F)(F)F)NC(C1CC(O)C(F)C1)=O c1(C(N2CC(NC(c3ccc(OC)c(N)c3)=O)C2)=O)cc2sc(C)cc2s1 C=CC1OCCC1C(=O)N(C1CC(C#N)C1)CC(=O)Nc1cc(C(=O)OC)ccc1C Cc1ncnc(C(=O)NCCCC2CN(C(C3(C)CC=CCC3)=O)CCO2)c1C n1(C(C)C)cc(OCC(=O)NC(C)CC2CN(C(C3CCO3)=O)C2)cn1 c1(C(N2CC=CC(NC(CC3CCC(C)CO3)=O)C2)=O)cc2ccccc2[nH]1 C1(NC(c2ncco2)=O)CCCCCC1C(=O)O c1(SC)ccc(CC(=O)Nc2ccc(OC(F)F)cc2)cn1 C1(C)(CNC(C2C3(CC(OCC)C3)C2)=O)CC(F)(F)CN1C(=O)CC1(C)CCC1 c1(SC)ccc(C(=O)NCC2(F)CC(CNC(C3CCCC3C)=O)C2)cc1 c1(OCC)ncccc1C(N1CCC(CNC(c2coc(C(C)(C)C)n2)=O)C1)=O C(=O)(C1CCCn2nccc21)NC(CN(C(C(C(C)C)NC(=O)OC)=O)CO)C C1(NC(Cc2c(C)cc(C)s2)=O)CCN(c2ccnc3ncnn23)CC(C)(C)C1 N1(C(CN(C2(C(F)F)CCC2)C)=O)CCCC(n2cncn2)C1 C(CCCCCCC(=O)N1CCC(NC(=O)C(c2cccc(F)c2)C)CC1)SC N1(C(Cc2scc(CN(C)C)n2)=O)CCC(n2cc(C3CC34CC4)nn2)CC1 N1(C(CN(CC#C)C(c2cncn(C)c2=O)=O)=O)CCC(F)(F)CC1 c1(C(C(=O)NC2CCC2)N(c2c(C)cccc2)C2CC2)c2c(nn1C)CCCC2 C(=O)(C1CCCc2nncn21)NC(C#N)CO c1(C(=O)NC(C)CNC(c2ccncc2Cl)=O)cc(Br)n(C)c1 CC1COCC(CC(=O)N(C)CCN(C(=O)C(O)(C2CC2)C2CC2)C)O1 C1(NC(CN(C2CCSC2)C(CC2CC(CC)C2)=O)=O)CC2CCC1C2 c1(C(N2CCCCC2c2ccc(C)o2)C(=O)NC)nc(O)sc1C C1(OC)CCC(C(=O)C(c2nn[nH]n2)NC(c2cc(CN)[nH]n2)=O)CC1 N1(C(C2N(C(C3CCC(=O)C3)=O)C3CCC2C3)=O)CCn2ccnc2C1 Cc1cc2c(C(N3CCC4CN(C(C5CCCC5O)=O)CCC34)=O)nccn2n1 Cc1nc(=N)[nH]cc1C(=O)NC1CCCN(C(C2(C3CCCO3)CC2)=O)C1 C1(C(N2C(C(N(CCCC)CC)=O)C=CC2)=O)C2CC(=O)CC12 O=C(NNc1ccc(Br)c(F)n1)NCC1CCCN1C(c1ccccc1)C1CCCC1 S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)NCCC(=O)NC1(C#C)CCCCC1 c1(CC)cc(C(N2CCC(OCCNC(=O)C(C)(C3CC3)OC)C2)=O)on1 c1(C(C)NCc2cccc(C(=O)OC)c2)c(C)oc2ccccc12 N1(C(C(CCCC)NC(c2nnsc2N)=O)=O)C2C=CCC1CCC2 c1(C(N2CCC(O)(CCNC(C3ON=C(C)C3)=O)C2)=O)cncc(Br)c1C Cc1ccc(C(N2CCOCC(NC(C3C(C)C3C)=O)C2)=O)c(O)c1C c1(C(N2C(CN(C(C(CC)(C)C)=O)C3CC3)CCC2)=O)[nH]c2ccccc2c1Cl N1(C(C=CSC)=O)CCC2(CCCCC2NC(c2ccsc2C(F)F)=O)C1 C(C(C)(O)CC(=O)N1CCC(C(=O)NC2(C(F)(F)F)CC2)C(C)C1)OC C1(S(N)(=O)=O)(C(=O)NCC(CNC(C2(C)N(C)CCC2)=O)O)CCCC1 C1(CCNC(CCC(=O)OCC)=O)CCN(C(=O)Cc2cnc(C)[nH]2)C(C)C1 C1(C(=O)O)C(N)C2CCCCC12.C1(CN(C)C)(NC)CCCCC1 C1(CC=C)(C(=O)NCC(CC)NC(=O)COC2CC=CC2)CCOCC1 C1(CNC(C2(CNC(C=CC(C)(C)C)=O)CCC2)=O)CC2CCCC2C1 C(=O)(CCCCCC(C)O)NC1(CNC(C(CC)n2cccn2)=O)CCCCC1 Cc1cc(O)ncc1C(=O)NC1(C(=O)NCCCC(C)(F)F)CC(CO)C1 CC(C)C(C)C(=O)Nc1cccc(C(N2CCC(C(C)C#N)CC2)=O)c1 C1(O)(CC(N2CC(CNC(CC(C)n3ccnc3)=O)OCC2)=O)CCCN(C)C1 c1(CC2(NC(C(c3cocc3Br)N(CCOC)C)=O)CC2)ccccc1Cl C1(C)(C(N2CC3C(CNC(c4n(C)c(Cl)cn4)=O)C3C2)=O)CC(C2CC2)=NO1 C(=O)(CC1=CCCC1)N(CC(C)CNC(C1(c2ccccc2)CCOCC1)=O)C C1(CNC(c2nc(CCC)oc2)=O)CCN(C(=O)CC2CC(N(C)C)C2)CC1 C(=O)(C(C(C)C)n1cnnc1)NCC(=C1CN(C(CC(C)C)=O)C1)F CCCCC(O)CC(=O)N1CC(O)CC1C(=O)N(C)Cc1cocn1 c1(CN(C2CCCNC2)CC)cccc2c1OCC2C.n12cc(nn1)CNC(=O)C2 C12(C(N(C(CC)C(=O)OC)C)=O)C(NC(C3(CC)CCCC3O)=O)C3CC1C2C3 CCCC(CC)CCC(=O)N1CC2CC(C(N3CCC(C)(CCO)C3)=O)CC2C1 C1(C(CNC(c2c(CC)csc2)=O)(C)C)CCCCN1C(=O)Cc1c(C)cnn1C N1(C(C(C)CC2CCC2)=O)CCC(C2CC2)C1C(=O)NC1(C)CCSC1 c1(CC)cn2c(C(=O)NC(C)CC(C)NC(C3CC(OC)C3)=O)cccc2n1 Cc1cc(C(=O)OCC(c2cn[nH]c2)=O)c(C)n1CC1CCCOC1 CC#CCCCC(=O)NC1C=CC(C(=O)NCC)C1.N12CCC(C1)OCC2 C(=O)(C(C)(C)S(C)(=O)=O)NCCC12C(CN(C(C3(CCC)CC(=O)C3)=O)C1)CC2 Cc1[nH]c(C#N)cc1C(=O)N(CC(=O)NC1(C)CCCCC1C)CC(C)C C1(NC(CC(C)C)=O)CCCOC1C1CCN(C(=O)C(F)=CCCF)CC1 N1(C(c2nn(CC)c(C)c2)=O)CCC2(CC1)CC2NC(=O)CN1CCCC1CO C(C)(C(=O)N(C)CC1(NC(=O)C(C)OC2CCCC2)CC1)NC(CCCC)=O S(=O)(=O)(c1ccccc1Cl)N1CCCC(C(=O)NC2CCOC2)C1 N(C1COc2ccccc21)C(C1C(C(=O)Nc2ccc(C)c(Cl)c2C)C1)=O N1(C(C(N2CCC(O)CC2)C)=O)CCC2(CC1)CN(C(=O)Cn1nccn1)C2 c1(C(N(CCNC(c2cc(OC)n[nH]2)=O)CC)=O)cc(C)c2c(O)n[nH]c2n1 C1(CC)CCN(C(=O)C(C)Cc2cnc[nH]2)C1CNC(=O)CC1CC2(CC2)C1 c1(CC(=O)NC2CCC(NC(c3cncs3)=O)C2)ccc2nc[nH]c2c1 C(CCC(C)(C)NC(C1CC1C(F)F)=O)NC(CC1C(CC)C1)=O c1(C(=O)NC2CC(C)(CNC(C(CSC)O)=O)C2)ccnc2ccc(Cl)cc12 CCCC(C)CC(=O)N1CCC(CF)(NC(c2cc3ccsc3s2)=O)C1 C1(CC(=O)NC(C2CCC2)C)CCCCC1NC(=O)C=Cc1nccs1 C(CC)(CO)N(C(CC1(N(C(C2C(CCC)C2)=O)C)CC1)=O)C1CC1CC C1(Cl)(C(N2CCCC(N(C(C3C(C)C3)=O)CC3CC3)C2)=O)C2CCC(=O)C12 C1(CCCC)CN(C(c2cc(C)c(C)[nH]2)=O)CCN1C(C1C2COCC12)=O c1(C(N(C(CCNC(C(CC(=C)C)C)=O)C)C)=O)cc(C#N)c2n1CCCC2 N1(C(CC2N(C)CCCC2)=O)CC2(CCN(C(=O)CC(F)(F)C(F)(F)F)CC2)C1 C1(C(N(CCNC(C(COC)(C)O)=O)CC2CC2)=O)CCCCS1(=O)=O c1(C(=O)OC)cn(CC(=O)NCC2CCC(NC(=O)C(C)NC=O)C2)cn1 N1(C(=O)CC2CCN2C(C2CCCC3(CC3)C2)=O)CCCN2CCCC2C1 c1(C(=O)NC2C(NC(CCCCC=C)=O)C2)ccc(Cl)c(C)c1O O=C(CCCCC(F)F)NCC1CC1CNC(c1cncc(C2CC2)c1)=O CCC(C)C(CC(=O)NC(C)CCN(C)C)NC(=O)CC1C=NN(C)C1=O CC1C(=O)N(C)CCN1C(C1(C)CCCN(C(c2ncc(Cl)cc2F)=O)C1)=O c1(C(=O)NCC2(F)CC(NC(C(CC)F)=O)C2)c[nH]c2ccc(F)cc12 c1(C(N2CC3C(NC(C4(C)CCCCC4)=O)C3C2)=O)cc(F)ccc1C#N CCC(CCCC(=O)NC(CO)C(C)O)NC(C1CC2(CC2)CN1C)=O c1(C(=O)NC(C(C)C)CCN(C)C(C2CC2(F)F)=O)c(Cl)ccnc1F C(=O)(CCCCCn1cnnn1)NCC(C(C)(C)C)NC(=O)COc1ccsn1 c1(C(=O)NCC(CNC(CCCC=C)=O)C)ccc(C)cc1Br c1(C(=O)NCCN(CCOC)C(C2CC(=C3CC3)C2)=O)ccc2ccncc2c1 N1(C(C(=O)NCc2ccccc2Cl)C2(C)CC2)CCN(c2ncccc2F)CC1 N1(C(CCc2c(C)cccc2)=O)CC(NC(=O)C(O)c2cnc[nH]2)CC(F)C1 CC(CC1CCCO1)C(=O)NC1(CCNC(=O)CC2(C(F)F)CC2)CCC1 N1(C(CCCOC)=O)CC2CCOCC2(NC(c2cc(C(C)=O)cn2C)=O)C1 N1(C(C=CC(C)(C)C)=O)CC2(CCOCC2)C1C(=O)NCCNC(=O)N(C)C N1(C(C(=O)NC(C)C)CC2CCOC2)CCOC2CS(=O)(=O)CC12 C1(C(=O)NCC(C(=O)N(C)Cc2ccccc2)OCCOC)C2CC3C(C2)C13.OC C#CCN(OC)C(=O)C1C2CCN(C(=O)CCc3ccncc3)CC12 C12(C(=O)NC34C(C)OC(CNC(C5CCOCC5)=O)(C3)C4)CCCCC1C2(F)F C(=O)(CC(CSC)NC(=O)C(O)CSC)NCC(CC)(C)O Cc1n[nH]c(C)c1S(=O)(=O)N1CCC(O)C(Nc2ncnc3ccccc23)C1 N1(C(C2(COCC)CC2)=O)CC2CC2C1CNC(=O)CCc1ncc(C)[nH]1 CCCC(C)C(=O)NC1CN(C(=O)Cc2ccnc(OC)c2)CC1C C(=O)(CCP(C)(C)=O)NC1C(C)CN(C(c2cc(-c3ccc(Cl)cc3)no2)=O)C1 C12(CNC(=O)CC(F)F)CN(C(C3CCCC4(CCC4)O3)=O)CC1CCO2 c1(NC(C2CC(O)CN2C(=O)Cc2ccc(O)cc2)=O)c(F)ccc(Cl)c1F C1(NC(CNC(C)=O)=O)CCN(C(C2CCCN2C(=O)C(C)C)=O)CC1O c1(OC)cnccc1C(=O)NC12CC(C1)N(C(=O)CC1CCCCC1O)C2 C1(C(=O)N(C(C)Cc2cccs2)C2CC2)C=CC(NC(=O)C(CO)N(C)C)C1 C1(N(CCc2c(C)ccnc2)C)CCc2cc(Br)ccc2C1 c1(C(N2C(C)(C)C(CC(=O)NC3CC34CC4)CC2)=O)cccc(S(N)(=O)=O)c1 C(C(CC(C)C)C(=O)NC1CC12CC(NC(c1cccc3[nH]ncc13)=O)C2)OC c1(C(N2CC(C(N3CCCC(O)CC3)=O)C2)=O)ccc2ccccc2n1 c1(CN(CCN(CCC(c2ccccc2)C)C)C)c[nH]c2cccnc12 N1(C(c2c(C)sc(O)n2)=O)CCC2(CCCCC2NC(=O)CC2(N(C)C)CCC2)C1 C1(CC)(Nc2nc(Cl)oc2C)CCN(C(c2ccc(Cn3ccnc3)o2)=O)CC1 C(=O)(C1=CCCCO1)NC1C(CNC(=O)Cn2cc(-c3ccccc3)cn2)C1 Cc1cc(C(N2CC(NC(=O)CCCCBr)C(O)C2)=O)nn1C C1(CNC(c2cc(CCO)on2)=O)CC(O)CN1C(=O)CC1COCCO1 CC(C)C(F)C(=O)NC(C)(C)CNC(C1OCCO1)=O c1(C(N2CC(C)(C)C2C(C)C)C(=O)NCCSC)nn(C)c2c1CCC2 C1(C(N(C2CCS(=O)(=O)C2)CC(CC)N(C)C)=O)CCCCC1C(C)(C)C N1(C(c2cnn(C)c2C#N)=O)CC=C(CC(=O)NC2CCOC2(C)C)CC1 c1(CNC2CC(NC(CCC3CCC(C)O3)=O)C2)ncccc1Cl C1(C)(C(N(CC(O)CNC(=O)CC2(C(F)(F)F)CCC2)CC)=O)CCCN1C N1(C(CC2(CC)CCOCC2)=O)CC(C)(C)CC1CNC(c1n[nH]cc1OC)=O c1(C(N2CC(NC(=O)C3CC3)C(CC34CCC3C4)C2)=O)ccc(C2CC2)cc1 C=CCC(CC)C(=O)NCCOCCNC(=O)Cc1c(C)ncnc1C C(=O)(C(C)CC(C)C(C)=O)NCC(CC(=O)NC(CC)CCO)O C=CCC(C(=O)NC1CCC(CNC(=O)C(C)COC)CC1)C(C)C N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(C)(C)C(NC(c2cnc(O)cc2C)=O)C1 C1(NC(CCS(C)=O)=O)CC2CC(NC(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 C1(CC(=O)NC2CCC(NC(C3C(COC)C3)=O)CC2)CCC2(CCCC2)CC1 Cc1ccc(NC(=O)C(=O)N(C)CC2COC(C)C2)c(C)c1 c1(C(=O)NCC(C)N(C(c2n(C(C)C)cnc2)=O)C)ccc(CO)nc1 c1(C(=O)NC2CC(N(C(=O)C(O)CC3CC3)C)C2)c(F)cccc1[N+](=O)[O-] O(N1CCC(CC(N2CCCC(CCNC(=O)C(C)(C)F)CC2)=O)CC1)CC C1(O)(CC#C)CC(NC(c2ccc(NC(=O)CC3CC3COC)s2)=O)C1 C1(CN(C(=O)C(c2ccccc2)O)C)CC(F)CN1C(=O)Cc1ccc(Cl)cn1 N1(C(Cc2snc(C)n2)=O)CCC(NC(c2ccc(F)c(Cl)n2)=O)C(F)C1 C1(NC(CCC(=O)N(C(C)C)C)=O)CC(F)(F)CC1NC(C1CC2(CC2)CO1)=O N(C)(C(=NCC(F)F)NCC1CCC2(COC2)O1)Cc1c(C)c(Cl)ccc1 c1(NC(C2C(C(N3CC(N(C)C)C3)=O)C2)=O)cc2ncccc2[nH]1 n1(CC)cnc2nc(N3CCC(S(N)(=O)=O)CC3)nc(NCC(C)(C)CSC)c12 C(=O)(CC(C)(O)CNC(=O)COC(=O)C(C1CCCNC1)C)OC C(c1ccc(C)o1)=CC(=O)N(C(C(=O)NC(C(=O)NCCC)C)C1CC1)C c1(C(=O)NC2C(CNC(c3ccc(CO)c(F)c3)=O)C2)ncnc(O)c1Cl Cc1[nH]nc(CN2CCC(C(=O)N(C)CC3(c4ccno4)CC3)C2)c1F N1(C(C2(COC)CC2(F)F)=O)CCOC(CNC(C2CC=CC(O)C2)=O)C1 C1(C(N2C(CN)CC(C)(C)C2)=O)CC12CCN(CC(N)=O)CC2 c1(C(N)=O)cc(C(=O)NCc2nocc2C(=O)NCC2C3CCCC23)n[nH]1 n1(CC(N2CCOCC(NC(c3nc(CC)oc3)=O)C2)=O)c(C)cc(O)cc1=O C1(NC(C2CCC(=O)NC2)=O)CCCCCC1C(=O)N.N1(CC=C)CC2CC2C1 C1(NC(C(C)SC)=O)CCN(C(=O)CCn2c(C)csc2=O)C1(C)C C(=O)(CC1=CCN(C(=O)C(C)(CC)CO)CC1)N(CCCC=C)CC c1(-c2nnc(NC(C3CCC3F)=O)s2)ccc(F)cc1 c1(C(=O)NCCOCC(=O)NC(C2CCOC2)C)cc(Cl)ns1 CCC(CC(=O)N1CCC(CC(=O)N2CCC2)C1)C(C)(C)C S(=O)(=O)(c1cccc(=NCCC(C)CCCC)[nH]1)NCCOC c1(C(C)C)nccc(=NCC2CCCN(C(=O)CN3CCC(C)(C)C3)C2)[nH]1 c1(C(c2ccccc2)NC(=O)NCc2occ(CC)n2)cc(Cl)cnc1F C1(N(C(COCCCC(C)C)=O)C)CC2CC1N(C(c1cc(Cl)ns1)=O)C2 C1(CN2CCC(C(N(C)C)=O)CC2)CC2(CCC2)CCO1 N1(C(CCCC)=O)CCN(CCCN(C(C2CCN(CC(C)C)CC2)=O)CC)CC1 C12(CNC(Cn3ccc(C)n3)=O)CC(CNC(=O)CC3CC=CC3)(CO1)C2 C1(CNC(C(C=CC)O)=O)CCN(C(c2nc(C)ccc2C)=O)C1(C)C C12(NC(CSC)=O)CCN(C(=O)C(C)(C)c3cccs3)CC1C2 c1(OC)cc(F)c(F)cc1CN1CCC(CC(=O)Nc2ccc(C)c(F)c2)CC1 n1(CC)cc(CC(=O)N(CCCOCCNC(=O)CC2CCCC2C)C)cn1 Cc1cc(N)ccc1C(N1CCCC1CNC(c1ccsc1C(F)(F)F)=O)=O C1(C(=O)NCC(F)Cl)CCCCCCN1C(=O)Cc1cnoc1 C=CC(O)C(C)(C)C(=O)N1CC2C(C(=O)N(C3CCC(O)CC3)CC)C2C1 C1(NC(Cc2cc(C)ns2)=O)CCC(C)N(C(=O)Cn2nccc2C)C1 C1(CNC(c2c(OCC)cncn2)=O)CCN(C(=O)CCCCCSC)C(C)C1 c1(C(=O)NCC=C2CCN(C(COCCC)=O)CC2)ccc(C2=CCCC2)cc1 N1(C(c2c(CC)nn(C)c2Cl)=O)CCN(C(C2CCCC(C)C2)=O)C2(CCC2)C1 N1(C(Cc2c(C)nc(S)s2)=O)CCC2(CCCC2NC(C23CC(C)(C2)C3)=O)C1 c1(CC(N2C(C)CC(CNC(C3(CC=C)CC3)=O)C2)=O)c(C)nn(C)c1C C(=O)(CS(=O)(=O)CCO)N(C1CCC(NC(CSCCC)=O)CC1)C C1(NC(CCNC2CC2)=O)CCCC(OC)C1.C12CC(C1)C(=O)N2CC S(=O)(=O)(c1cccc(=NC2CC(CC#N)C2)[nH]1)NCC1CC(C)(C)OC1 n1(CC)nc(C(=O)NC2CN(C(C3(CC(C)C)CC3)=O)CC2O)ccc1=O C=C(F)C1(CC(N2CCC(F)(C(=O)NOC3CCOCC3)C2)=O)CCC1 N1(C(CCC#C)=O)CCC2C(CCN2C(c2cn3ccc(C)cc3n2)=O)C1 c1(C(N2CC3C(NC(=O)Cc4cncs4)(C3)C2)=O)cccc2ncccc12 N1(C(Cc2c(C)nc(SCC)s2)=O)CCN(C(=O)C(CC)=CC)C(C)CC1C CC(C)CC(CNC=O)CC(=O)NC1CN(C(C2CCCC23CC3)=O)CC12CC2 c1(OC)ccc(C(=O)NCC(O)CNC(C2COCC2C(F)(F)F)=O)cc1N C1(NC(c2cc(C)on2)=O)(CNC(c2cnc(S)n2C)=O)CCCCC1C C1(CC(N2CC(C(=O)NC3C(C(=O)OC)C3)C2)=O)CC2(CCC2)CO1 C1(F)(CNC(=O)CC2CCOC2)CCC(CNC(=O)C(=O)N2CCC2)C1 CC1CCc2[nH]c(=NC3CCOCC3)nc(N3CCC(C4CCC4)CC3)c2C1 N1(C(c2cc(C(=O)OC)no2)=O)CCC(O)(C(C)NC(C2CCSCC2)=O)C1 N1(C(CCOC)=O)CCN(C)C(CNC(=O)CCC(C)OCC)C1 CCC(C)C(C(=O)NC(C)CN(C(=O)CCCc1nnc(C)s1)C)NC(C)=O c1(OC)ccc(C(=O)NCC(CO)NC(C2CC2c2ccc(Cl)nc2)=O)cc1O Cc1cc(C(N2CCCC2CC(N2C3CCC2CC3)=O)=O)cc(C)c1C N1(C(CCSCCCC)=O)CCC2C(CCCN2C(=O)CCN2CCCC2)C1 c1(OC)nccnc1C(=O)NC1CC2(C1)CC2C(=O)NCCCS(C)=O C(=O)(CC(CNC(=O)C(C(C)C)N(C)C)C1CCC1)NC(CC#C)(C)C C(=O)(CCCN(C(=O)CCc1nncs1)C)N(C(CC)COC)C c1(CNC(CCn2cc(-c3cccc(OCC)c3)nn2)=O)cc(OC)nc(Cl)c1 CCC(C)C(C(C(=O)NC1CCCC1)N(C)C(C)C)OC.C1(C(=O)N)(C(C)C)CC1 C1(C)(OC)CCCN(C(=O)C(CNC(c2ncccc2O)=O)CC(C)C)CC1 CS(=O)c1cccc(C(N2CC(F)(F)CC2CNC(c2nc(Cl)cs2)=O)=O)c1 C(CCN(C)C(c1cc(C)cs1)=O)(C(C)(C)C)NC(C(CCSC)O)=O N1(C(Cc2cn(CC)nc2)=O)CCC2(CC1)CC2NC(C1CC1c1cnc[nH]1)=O c1(NCCCCC(=O)NCC2(C(=O)OC)CC(=C)C2)cncc(Cl)c1 c1(C(N2CC(NC(C(C)(F)F)=O)C3C2C3)=O)cnc2[nH]ccnc1-2 C=C1CC(C(=O)NCCCc2ccccn2)(CNC(C2CS(=O)(=O)C2)=O)C1 c1(C(=O)NC2CCCN(C(c3n[nH]cc3F)=O)CC2)ccc(Cl)c(Cl)c1O N1(C(c2nn[nH]n2)CC)CCC(CSC)CC1 N1(C(C(COCC)C)=O)CCC(O)CC1C(=O)NOCc1ccc(O)cc1 S(=O)(=O)(c1ccc2c(c1)CCCN2)N1CC(C2CC(=O)NC2)OCC1 N1(C(c2ncn(C(C)C)c2)=O)CCC2(C(=O)N3CC(O)CO3)CC2C1 S(=O)(=O)(c1ccc(CCC(C)(C)O)cc1)NC(C1CN(CCS(C)=O)C1)=O C1(N(C(C(CC#C)C)=O)C)CCCCN(C(c2ccc(OC)nc2Cl)=O)C1 C1(CCC(=O)N(CCC)CCC)CCCCN1C(c1[nH]ccc1COC)=O c1(C2(CNC(N(C)Cc3c(OC)cccc3)=O)CCC2)ccc2c(c1)OCO2 N1(CC(N2CC(NCC3CCS(=O)(=O)C3)C3(CC3)C2)=O)CCCCCC1=O N1(C(c2c(C)cccc2)=O)CC(CO)C2(C1)CN(C(C1CC(N(C)C)C1)=O)C2 c1(C(N2CCC(C(F)(F)F)C(NC(=O)C3CC3)C2)=O)cnc2ccccc2c1OC CC(C)CC(CNC(=O)C(C)Oc1ccccc1)NC(c1cccnn1)=O N1(C(CC(CNC(=O)C=C2CCCCC2)OC)=O)CC2CCC1C(O)C2O C1(CNC(CCc2cn(C)nn2)=O)CC12CCN(C(c1sccc1Cl)=O)CC2 CC1CCC(C)(C(=O)NC2CCCCC2CC(N2CCC(CF)CC2)=O)CC1 C(=O)(C1CCCc2ncccc21)NCCN(C(=O)CCCS(N)(=O)=O)CC CCC(F)(F)C(=O)NCCC1(NC(=O)CCc2cccc(O)n2)CCC1 C12(CNC(C=Cc3ccc(C)s3)=O)CN(C(=O)CC3CCCCC3)CC1CCO2 c1(C(=O)NCC(CNC(=O)C=C(Cl)Cl)C(F)(F)F)cc2ccccn2n1 Cc1sc2cncn2c1CNC1CCNC(C2CC2)C1 n1(CC(=O)NC23C(CN(C(C4(CC)CCC4)=O)C2)C3)ncc2cccnc12 CCC(CC(=O)N(C(CNC(c1cn(C)nc1C(F)F)=O)C1CC1)C)C1CC1 C1(CC)C(N=c2[nH]c(CCC(C)C)cs2)CCCN1 c1(CNC2CN(C(c3ccc(OC)c(Br)c3)=O)CC(C)C2)ccc(F)c(F)c1C c1(C(N(CC(=O)NCC(C)(CO)CO)CC2CC2)=O)ccc2nccn2c1 c1(SCCC(=O)NC2C(NC(CN3CCC(C)CC3)=O)CC2)ccc(F)c(F)c1 Cn1cc(-c2cn(C3CCN(C(C4CCC(F)(F)C4)=O)CC3)nn2)ccc1=O C12(C(N3CCCC(C(=O)NC(CC=C)CC)C3)=O)CC(C)(CCO1)C2 c1(OC)nn(C)cc1CNC(=O)C(Cn1ccnn1)NC(=O)C(C)CC1CC1 C(=O)(CCCC(=O)NCCCC1CCOCC1)OC(C)(C)C C1(C(C)C)(C(=O)NC2COCC2CO)CCN(C(c2cncs2)=O)C1 C1(CC(=O)NCC(C)(CO)NC(C(N2CCOCC2=O)C)=O)CC(=O)NC1=O c1(C(N2CC(OC)C3C(C2)CC3)=O)cccc2cn(C)nc12 c1(CC)cc(C)ccc1C(=O)NC1CCCC1CNC(=O)CC1CC(O)C1(C)C N1(C(COc2cn(C)nc2)=O)CC2C(CCNC(=O)CC3CCOC3)C2C1 Cc1ccnn1C(C)C(=O)NCC1(C(=O)NC2(CF)CCC2)CCCO1 C1(C(=O)NCCC(=C)CNC(=O)C(F)CC(C)C)CC2(CCCCC2)S1(=O)=O CCCCC(CNC(=O)CCCCC)NC(c1snnc1CCC)=O NC(=O)CC(C(=O)N1CCC1C1CCCC1)NC(C1CCC2(CCC2)C1)=O CN1CCC2(CCN(C(C3CCC(CNC(C4(C)CC5CC5C4)=O)C3)=O)C2)C1 N1(CCC(=O)N(C(C)C)CCNC(C2(Cl)CC2(F)F)=O)CCCS1(=O)=O c1(SCC(=O)NCC(C2CC2)NC(C(F)=CCC)=O)nnc(S)s1 C1(C(=O)Nc2cnc(CC)nc2)CCc2cc(S(N)(=O)=O)ccc2O1 CCC(C(=O)N1CCC1C(=O)NCCc1cnc[nH]1)N1CCCC1=O CC(C)(CO)C(c1ccccc1)NC(=O)N(CCO)Cc1cscn1 C1(C(C)C)(CNc2ccc(-c3nnnn3-c3ccccc3)o2)CC(C)(C)C1 Cc1cc(C(=O)NC2CCCN(C(C3(C)CC4(CC4)C3)=O)C2)ccc1O Cc1cccc(CC(=O)NCCNC(c2n[nH]c3c2COC3)=O)c1F Cn1nc(C(=O)NC(C2CCN(C(=O)CN3CSCC3=O)C2)(C)C)cc1C(F)F c1(C(N(C(CN(C(c2c(C)cc[nH]2)=O)C)C)C)=O)ccc(C(N)=O)nc1 C(=O)(C#CC1CCCC1)N1CC(NC(Cc2c(C)nn(C)c2Cl)=O)C(C(F)F)C1 CCC(C)C(CC(=O)NCCC(C)C(C)(C)C)NC(C1CCCC(=O)CC1)=O c1(OC)c(CN2CCC(F)(CNC(c3ccncn3)=O)C2)cccc1Cl c1(C(N2CCCC(NC(C)=O)C2)=O)nc(C)ncc1Br.C1(=O)CCCCN1 Cc1ccc(Br)c(C(=O)NC2CCN(C(C3CC=CCC3)=O)CC2(C)C)c1F c1(C(N2C(C(=O)OC(C)(C)C)CC2C)C(=O)NC2(C)CC2)cc([N+](=O)[O-])sn1 N1(C(C(CCO)N(C)C)=O)CC(C)(C)OCC1CNC(c1cc(C(F)F)no1)=O c1(C(CNC(CC)=O)NC(c2cc(C(=O)OC)nn2C)=O)cccc(C)c1 C1(NC(c2cc(C)no2)=O)CCC(C)N(C(=O)COc2ccc(F)cc2Cl)C1 CC1(C(=O)NCCOCCNC(c2cn(C(C)(C)C)nn2)=O)C=CCC1 C(C(=O)N1CC(Cc2cn(Cc3ncccn3)nn2)C1)(C(C)(C)C)OC(C)C c1(OC)ccc2[nH]c(=NC(=O)N(C)C)[nH]c(=NCCn3ccnn3)c2c1 c1(CC)oc(C(=O)NCC2CCC(NC(c3cnn(C)n3)=O)C2)cc1C C1(NC(c2cccc(CC)n2)=O)CCCN(C(=O)CC(CC)C2CCC2)C1C C(=O)(CCS(C)=O)N(C1CCN(C(=O)C=Cc2cncn2C)C1)CCC C(=O)(C1=CCS(=O)(=O)C1)NCC(C)NC(=O)COc1cc(F)cc(F)c1 c1(CCC(=O)NC(CNC(C2(C)C(C)(C)C2)=O)C2CC2)ccc2c(c1)OCO2 N1(C(C(C)OCCOCC)=O)CC(O)(CCNC(=O)C(C(=O)OC)N(C)C)C1 C1(C(=O)NCC2N(C(C(CC#C)(C)C)=O)CCC2)CN2CCN1CC2C C(=O)(NNc1ccc(F)cc1I)NC(CCN(C)C)C(=O)N1CCOCC1 N1(C(C=COCC)=O)CC2CCC(C3CC3)(C2)C1 c1(CN2CCC(CCCCCNC(C=C(C)C(C)C)=O)CC2)ccc(O)cc1F c1(C(=O)NC2(C)CN(C(C(C)CF)=O)C2)ccc(N2CCCC2)cc1 CC(c1cccs1)=CC(=O)NCCC1CSCCN1C(C1CCC(C)O1)=O Cc1cccc(C(=O)NCC2CN(C)CCN2C(C2CC23CCC3)=O)c1N N1(C(C(CC)N(C)C)=O)CCC(C(=O)NCCCN2CCOCC2=O)(CC)CC1 N1(C(c2c(OC)cccc2)=O)CCC(NC(=O)Cc2cn(C)nn2)C(C)(C)C1 c1(C2(C)CC2)cc(C(=O)NC2CCCC2NC(=O)CSc2cc[nH]n2)no1 N1(C(C=CCCC)=O)CCN(C(c2csc(C)c2N)=O)C(c2ccncc2)C1 c1(C(=O)NC(C(C(C)C)NC(=O)C2=NNC(=O)CC2)C)cnc2ncccc2c1 C#CCCC(C(=O)NCC(C1CCC1)OC)NC(C1CCCCO1)=O C1(C(C=C(c2ocnc2NC(=O)CCC)C)=O)CCCCN1C(=O)OCC N(C1c2ccccc2CC1Br)C(=O)CN1CCSCC1 c1(C(N2CC3CCC2CN3Cc2c(F)cncc2Br)=O)cc(Br)cc2cc[nH]c12 C=CC1(CC(=O)NC2CN(C(=O)C(C3CC3)C3CC3)CC2C)CCCCC1 N1(CC(=O)NC(C)C(F)(F)F)CCN(C2CC(c3ccc(Cl)cn3)C2)CC1 C#CC1(N(C(=O)C2=NOC(C(C3CC3C)=O)C2)C)CC(F)(F)C1.C(=O)(CN)NC CC1CN(C(=O)C(c2ccccc2)C)CCN1C(c1cc(Br)n[nH]1)=O c1(C(=O)NC(C)CNC(=O)C(C)NS(C)(=O)=O)occc1Cl Cc1cccc(C(C)NC(=O)CNc2cccs2)c1 Cc1ccc(N(C(=O)C(C)CN(C(=O)C(C)n2cncn2)C)C)cc1C C1(NC(=O)CC2CC2)CCCCC12CCN(c1ncnc3c1COC3)C2 [N-]=[N+]=NC(CCC(N)=O)C(=O)NCC1CCCCN(C(=O)C2=CCSC2)C1 C1(NC(CC(CC)N(C)C(C2CCCC2O)=O)=O)CCCCCC1C N1(C(CC(CC)O)=O)CCCC2C1CCN2C(c1cc(I)ccc1Br)=O c1(-n2c(C)nnn2)ccc(C(=O)NC(C)CCNC(=O)C(C)n2cncn2)cc1 Cc1cnc(Cl)cc1C(=O)NC1CN(C(=O)CO)CC1O N1(C(c2nc(OC)oc2)=O)CC(O)CC1CCCNC(=O)Cn1nc(C)cc1C n1(CCNC(c2n(CC)nnn2)c2cnc(C(F)F)s2)nc2ccccn2c1=O Cc1ncc2n1CCC(C(N1CCC(N3CCC(NC(N)=O)CC3)C1)=O)C2 Cc1cc(I)c(F)cc1NC(C1CCCC(NCc2cccc(CO)n2)C1)=O c1(CC(=O)NCCOCCNC(=O)C(O)C(F)(F)F)ccc(O)c(F)c1 C=CC(CC)CC(=O)NCC1CCCCN(C(=O)CN2CCN(C)CC2)C1 C1(NC(CCSCCC)=O)CCC(C)(CNC(=O)CCc2cnn(C)n2)CC1 N1(C(C2(F)CCC(C)CC2)=O)CCC2(C1)CN(C(=O)Cc1ccsc1Cl)C2 c1(-c2c(C(N(C)CCNC(C3CC3F)=O)=O)cccc2)cccc(C#N)c1 C1(NC(Cc2nnc(C)o2)=O)CN(C(c2cncc(Cl)n2)=O)CC1F C1(C(N2CC(O)(C(C)NC(c3cc(C4CC4)no3)=O)C2)=O)CN(CP(C)(C)=O)C1 C(=O)(CC(C(C)C)C(C)C)N(C1CCCN(C(C2(OC)CCOCC2)=O)C1)C c1(CC)cnc(N2CCC(C)C2CNC(=O)C(c2c(C)n[nH]c2C)C)nc1 C=CCC(CCCCC)C(=O)N1CC2CC(CNC(=O)CCc3cnco3)C2C1 c1(CC(N2CCC(N(C(=O)CCN3CCOC3=O)C)C2)=O)ccc(F)nc1 N1(C(CC2CCC(NC(COCCCC(C)C)=O)CC2)=O)CCCCCC1C CC1CN(C(C2(Oc3ccccc3)CCCC2)=O)CC(NCC2CCCC3CC23)O1 N1(C(C(=CC2CCCC2)C)=O)C2CC1CN(C(=O)C(C)n1cccn1)C2 C1CN(CCO)C1.C(C(=O)NCCNC(=O)CNC(=O)NC)OCC c1(C(N2C(CNC(c3c(C)cccc3)=O)C(C)CC2)=O)c(Cl)ccc(O)c1Cl c1(CC(C(=O)NCCC(=C)CNC(c2cnoc2C)=O)C)c(C)nn(C)c1C C12(CN(C(CC3(C)N(C(CC4CC(N(C)C)C4)=O)CC3)=O)CC)CCC(CC1O)C2 N1(C(c2nccc3ccn(C)c32)=O)Cc2n[nH]cc2CC1C(=O)O C1(C(N(CC)CC)=O)C=CCNCC1.c12ccccc1c2=O c1(C(=O)NC(C)CNC(=O)CCP(C)(C)=O)sc2cc(F)ccc2c1Cl N1(C(c2ccc(F)c3c2CNC3)=O)CCS(=O)(=O)CC12CNC2 CC1=NN(C)C(=O)C1CC(=O)NCC=CCNC(c1sccc1CC#N)=O c1(C(=O)NCC2CC(C)N(C(c3cc(O)nc(O)n3)=O)C2)cn2c(n1)CCCN2 C(=O)(C1=C(C#N)CCC1)NCC(C)NC(CCc1c(C)noc1Cl)=O c1(OCCCC(=O)NCC2C(NC(C3CC3(Cl)Cl)=O)C2)ccc(F)cc1F CCC(CC)C(F)C(=O)N1CC=CCC1C(=O)N(C)OCC(F)(F)F CN1CCC(CC(=O)NCCOCCCNC(=O)CO)C1=O C12(NC(CCNC(=O)OC)=O)CCN(C(c3ccc(CC4CC4)s3)=O)CC1C2 c1(NC(C2CCN(C(c3cc(OC)n[nH]3)=O)C2)C)ncnc2cnccc12 c1(CC)ncncc1C(=O)NCCCCCCN(C(=O)Cc1cc(C)on1)C CCCC(C(=O)NC1CC2CN(C(=O)CCOC)CC2C1)C(C)C c1(OC)cc(F)c(C(N2CCCCC2c2nnc(C3CCOCC3)o2)=CC)c(F)c1 CCCC(CC)CC(=O)N(CCNC(c1cc(Br)cn1C)=O)CC C1(C(=O)NCC(CNC(CCCCOC)=O)O)CC2CCC1CC2 C1(C(=O)NC(c2cccc(C)n2)C)CC2(CC2)CN1C(c1csc(C)c1)=O C#CCC(O)C(=O)N1CCC(NC(=O)C(C#N)CC)C1 c1(C(=O)NCCCNC(C2CC(C)OCC2)=O)cccc(Cl)c1[N+](=O)[O-] CC1CN(C(=O)CCn2ccnn2)CC(C)N1C(C1CC2(CCC2O)C1)=O CC1CN(C(=O)CNc2cccnc2)CCC1N(C)C(c1coc2c1COC2)=O c1(C(N(CC)CC2CCCN2C(=O)Cc2cc[nH]n2)=O)csc2ccc(F)cc12 C1(N(C(CC(c2c(C)n[nH]c2C)C)=O)C)CN(C(c2occc2F)=O)CC12CC2 c1(C(=O)NCC(CNC(C2CC(N(C)C)C2)=O)O)ccc(C2CC2)nc1 C(=O)(CCCCCC)NCC(C(=O)NC(C#CCC)(C)C)O C(N=C(NCC(C)(C)C1CCC1)NCC1(C(F)(F)F)CC1)C1(C)CC1 N1(C(CC2(C)CC2F)=O)CC2CCC1C(NC(c1cc(F)cc(F)c1N)=O)C2 N1(CC(=O)NC(COC)C)CCCC(N(C(=O)CCC(C)(C)C)C)C1 c1(C(=O)NC(CCC)CNC(=O)C(C)CCOC)nc(C)ccc1F N1(C(CCCCOC)=O)CCC2(CCC2)C(NC(=O)C(C)CN2CCOCC2)C1 C(C1=NOC2CN(C(c3cccc(N)c3F)=O)CC12)NC(c1ccc(SC)s1)=O C1(C(N(CCCCCO)C)=O)CC2(CC2)CN1C(=O)Cc1cncnc1 c1(CNC(C2(c3cn(CC)nn3)CCOC2)=O)[nH]nc(OC)c1Cl.C1CC(C)(C)C1 c1(C(=O)NCCCCCNC(C2C(CCC)CCC2)=O)ccnc2c1nnn2C C1(OC)CCC(C(N2CC(NC(=O)CC(=O)NCC3CC3)C(C)C2)=O)CC1 c1(OC)cnncc1C(N1CCCC(C(C)C(=O)N(C)Cc2scnc2C)C1)=O C(=O)(CC(C)CC(F)(F)F)NC1CN(C(C2(C(=O)NC)CC2)=O)CC1O CON=CC(=O)NC(C(=O)NC(c1cncn1C)CO)C1CCOC1 CCC1=C(C(=O)N2CCC(C(=O)NCCN=[N+]=[N-])C2C(C)C)CCCO1 N1(CC(=O)NC(C)CNC(=O)CCN2CCC(F)C2)CCCCCCC1=O CC1=CCC(C)(C(N2CCCC(O)(CCNC(c3cnc(S)[nH]3)=O)C2)=O)CC1 c1(C(N(CCC(=O)N(CCOCC=C)C)C)=O)ncc(N)cc1C N1(C(C(COC)N(C)C)=O)CCC(O)(CCNC(=O)C(C)c2cccs2)CC1 C1(CC(N)=O)CCCN(C(=O)C(CCF)NC(=O)C2=NOCC2)C1 C(=O)(C(CC(C)C)ONC(C1CCS(=O)(=O)C1)=O)NC c1(C(=O)NCC2(F)CC(CNC(C3(O)CC3)=O)C2)coc2c1NC(=O)CCC2 Cc1ccc(Br)c(C2(C(=O)OCCCCC3CCC(C)(C)CC3)CCCC2)c1 c1(C(=O)NCCOCCCNC(CCCNCC)=O)cc(SC)ccc1Cl C1(C(=O)NCCCCCN(C(CN(C(C)=O)C)=O)C)C2CCC1(c1ccco1)C2 C1(C(=O)NC(C#C)(CO)CO)CN(C(c2ccccc2F)=O)CC1C1CC1 n1(CC(F)(F)F)nnnc1C(c1ccn(-c2ccccc2)n1)NCC1(C(N)=O)CC1 C1(CNC(c2c(CC)onc2C)=O)CC(F)(F)CN1C(c1cc(COC)cs1)=O N1(C(C2C(C(N(CC#C)C)=O)C2)=O)C2CCC1CN(C(c1cc(C3CC3)[nH]n1)=O)C2 CCCCCCCC(C(=O)NC1CCOCC1)N(C)OC(c1ccc(O)cc1)=O C(=O)(C(F)CC(CC)CC)N(C1CCC(NC(CNC(CC)=O)=O)CC1)C c1(C(=O)NCCC2(NC(c3cnc(C)[nH]3)=O)CCC2)[nH]nc([N+](=O)[O-])c1Cl C12(NC(C(C)NC(=O)C(C)(C)C)=O)CCCC1N(C(=O)CCC1OCCO1)CC2 C1(NC(=O)Cn2cccn2)Cc2ccccc2N(C(=O)C(F)C2=CCCCC2)C1 c1(C(=O)NCC2OCC(CNC(C=CCOC)=O)C2)cccc(S(C)(=O)=O)c1 CC1CN(C)CC1NC(=O)CNC(=O)C(c1ccccc1F)(F)F C1(C(N(C2CCCCC2)CCNC(C=CC=CCC)=O)=O)CCn2nccc2C1 c1(C(N2CCCC(C(F)(F)F)(NCC)C2)=O)cc(C)cc2nc[nH]c12 N1(C(CCC(C)C)=O)CCc2nc(O)cc(C(=O)NCC(C)C3CCC3)c2C1 n1(CC(CC(=O)OCC(c2cn(CC(CC)O)nn2)=O)O)ncc2ccccc12 c1(CC)cc(C(N2CCCC2CN(C(C2CCCCS2)=O)CC)=O)c(C)nn1 c1(C(N(CCC(=O)NCCC2CCCOC2)CC2CC2)=O)ncnc(O)c1F c1(C(=O)NCCCN(C(c2cc(C(C)C)no2)=O)CCO)ccn2c1CCCC2 c1(C=O)cnn2c1CCC2.C1(OC)CN(N2CCC(N3CC=CC3)C2)CC1C=O C(C(C)(C)COC(c1cc(C)n(C)c1)=O)(c1n(CC)nnn1)NC1CCSC(C)C1 NS(=O)(=O)c1cccc(S(=O)(=O)N2CCN(c3c([N+](=O)[O-])ncn3C)CC2)c1 C1(NCCNC(C)=O)CC2(CCOCC2)CO1.N1(C(C)C)CCOC1=O N1(C(C2(CCOC)CCC2)=O)CCC(C2CCN(C(=O)CC3CCCC3)CC2)C1 c1(C(=O)NC(CC(C)NC(C(CC#C)CC#C)=O)C)csc2ccc(OC)cc12 N1(C(c2c(C)nc(CC)s2)=O)CC2CC1CCN2C(=O)C(C)CC c1(C(=O)NCC(C(C)C)(C)NC(c2cnco2)=O)n[nH]c2c1CCC(C)(C)C2 c1(CNC2CC(C(=O)OC)C2)cccc2cccnc12 CN=c1[nH]nc(CC(=O)NC2CCCCC2NC(=O)CC2CCC2(C)C)s1 C1(CN(C(c2ccn(CC(F)(F)F)n2)C(=O)NC(CC)C)C)CCCS(=O)(=O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(CN1CCN(C(C=CC)=O)CC1)C C1(C)(NC(=O)NCCCNC(c2cn(C)nc2Br)=O)C2Cc3ccccc3C12 C1(CNC(c2nc(CCC)sc2)=O)C(OC)C(OC)CN1C(C1CCCOC1)=O C(CC(N)C(C)(C)C)NCc1c(N(C)C)ccnc1 Cc1cc(NCC2CC(NC(C3CC34CCOC4)=O)C2)n2ncc(C)c2n1 n1(CCOCC=C)c(N2CC(OCC)C(F)C2)nnc1-c1ccc(Cl)s1 C1(C(N2CCCC(NC(=O)C=Cc3cc[nH]n3)CC2)=O)CCc2cncn2C1 c1(NC(C2C=CC(NCc3cc(C)c(F)nc3)C2)=O)cccc(C#N)c1Cl C(CN=C(NCCc1ccco1)NCCN1CCCC1)c1ccc(C)nc1 CC1CC(C(=O)NC2(C)CCN(C(C3CCC(c4ccccc4)C3)=O)CC2)=NO1 Cc1ccc2sc(C(N3CC(NC(=O)C=CBr)CCC3C)=O)c(C)c2c1 Cc1cn2c(n1)C(C)CC(C(N1CCCC(CCNC(=O)CC3(C)CC3)C1)=O)C2 Cc1cc(C(N2CCCC(C(=O)N(C)Cc3nncn3C)CC2)=O)c[nH]c1=N C#CCCCCCCC(=O)NC1(CNC(c2cnco2)=O)CC2CCC1C2 C1(CNC(CCCC=C)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC1(F)CO Cc1cc(C)c(C(N2CC(NC(c3n[nH]cc3Br)=O)C(F)C2)=O)c(O)c1 C1(NC(C2C(Nc3c(SCC)cccn3)CC2)=O)CC(C)CN(C(=O)COC)C1 C1(O)(CC(=O)NC2C=CCN(C(C(CSC)(C)C)=O)C2)CCN(C)CC1 Cc1ncc(C(=O)NOCc2cn(-c3cc(Cl)ccc3Cl)nn2)cc1C#N c1(N2CCC3C(CSC)C3C2)nc(=NCC2(CC#N)CC2)[nH]c2cccc(F)c12 N1(C(CC=C(C)C)=O)CCC(F)(CNC(c2ncn(-c3cccc(F)c3)n2)=O)C1 C1(NC(C2N=C(C)SC2)=O)CCN(C(c2cc(C)ccc2O)=O)C1(C)C N1(C(c2cc(C(F)(F)F)ncc2Br)C(=O)NC)Cc2n[nH]cc2C1CO C=CC1(C(=O)NC2C=CCN(C(=O)COCC(c3ccccc3)C)C2)CCCC1 C1(C(=O)NCc2scc(CNC(=O)Cc3cnco3)n2)CC2(CC2)CO1 C(=O)(CC(C)(C)CC(F)(F)F)N1CCCC(C)(CNC(C(C)OCCC=C)=O)C1 n1(CC(=O)NCCC2CCN(C(CC=C=C)=O)C(C)C2)ccc(=O)c([N+](=O)[O-])c1 c1(OC)ccc(NC(c2ccc(C3CCC3)cc2)c2nnnn2CC(F)F)cn1 c1(C(C(=O)NCC(CNC(CSCC=C)=O)F)=O)cc(Cl)ccc1Cl C1(C(=O)NCc2ccc(SC)o2)CC12CCN(C(=O)C(C)NCC(C)C)C2 C1(NC(c2cccc(OCC)c2)=O)CC(NC(=O)CSCC)C12CCC2 C12(C(=O)NC(C)(CNC(=O)Cc3cnc[nH]3)Cn3cccn3)CCCC1CCC2 CCC(C#N)C(=O)NCC1CCC1C(=O)NCC1(C)CCC1 C1(C(N2CCCC(COC)C2)=O)N(C(C2CC3(CCC3)C2)=O)CCCC1(C)C C12(NC(c3cc(C(N)=O)co3)=O)CC3CCC(C1C2)N3C(C1CCOC1)=O N1(C(c2n(CC)ccc2)=O)CC2CCC2(CC(N2C(CO)CC2C)=O)C1 C1(C(=O)NCCCCN(C)C2CC2)CNC(=O)CN1C(=O)CC1CCCO1 C1(CC(=O)N(C2CC(NC(C(C)CC3CCC3)=O)C2)C)CC2CCC1CC2 c1(NC(C2CN(C(=O)Cc3cc[nH]n3)CCS2)=O)c(F)cc([N+](=O)[O-])cc1Br C1(OC)CN(C(C2CC(=C3CCC3)C2)=O)CC1C(=O)NOCCCO C1(C2CCC2)(C(N2CC(OCCNC(=O)CCc3cscn3)C2)=O)CCC1 N1(C(CC2(OC)CC2)=O)CCC(C)C(CNC(C2(CC(C)=O)CCOC2)=O)C1 c1(N2CCCC(C#C)(C)C2)ncnc2c1ncn2C(C)C(O)C(F)(F)F.C1CO1 c1(C(N2CC(CNC(CC=C)=O)OC3(C2)CCC3)=O)cc(C)nc2[nH]nc(C)c12 CC(C(=O)NCC1(c2ccccc2)CC(NC(c2cccc[n+]2[O-])=O)C1)C(F)F S(=O)(=O)(c1ccc(C(N2CC3CCC(CNC(C)=O)C3C2)=O)cc1)N(C)C c1(OC)nc(C(N2CC3CC3C2)C(=O)NCC2CCCO2)sc1C C(=O)(CS(=O)CC)NC(C#C)(C)C1CNC1 C(C(c1cccs1)=Cc1ccc(C(=O)O)cc1)C(=O)Nc1cccnc1OC(F)F C1(CNC(c2c(C)n(C)cn2)=O)CC2(CC2)CN1C(C1CN(C)CCO1)=O c1(C(=O)NC(c2ccc(C(=O)N(C3CC(O)C3)CCO)cc2)C)ccc(O)cc1 C(=O)(CC(F)(F)CC(=O)N1CCOC(CN(C(=O)C2=CCCOC2)C)C1)OC Cn1nc(C(=O)Nn2cc(C3CC4CCC3O4)nn2)cc1C1CC1.C12CN(C1)C2 N1(C(C(CC)N(CC)CC)=O)CC2CCN(C(c3cc(I)ccc3C)=O)C2C1.C(C)CC CC(C)(C)CCC(=O)N1CC(NC(=O)CCN2CCOCC2)CC(O)C1 C1(NC(c2nc(C(C)=O)sc2)=O)CCC(N(C(=O)C(C)C2CCC2)C)CC1 C12(C(N(C(CC(CC)C)C)C)=O)CC(CN(C(c3nsnc3O)=O)C1)C2 C(CCC1CCC1)(C(=O)N(c1ccncc1)CC(C)C)NC(CCC)=O c1(C(N(C(CCNC(c2n(CC)nnc2C)=O)C)C)=O)cc(F)cc(Cl)c1 S(=O)(=O)(CCCS(=O)(=O)C(F)(F)F)NC(c1cccc(CCC)c1)=O N1(C(CCC(=C)C)=O)CCCC(C2(NC(c3ccc(OC(C)C)nc3)=O)CC2)C1 c1(C(N2C(CNC(C=C(C)Cl)=O)COCC2)=O)ccc(F)c2occc12 Cc1cc(C)n2ncc(C(N3CCC(CF)(NC(=O)C4CC4)C3)=O)c2n1 CS(=O)(=O)CC(C(=O)O)N(c1ccccc1)CC1CC1 Cc1scnc1C(=O)NCC(C)(C)CN(C(=O)C(C)OCCC(C)C)C N1(c2ccccc2)CCCC(SCc2noc(C3CCCCC3)n2)C1 c1(C(N2CCC(NC(c3cc(C)c(Cl)s3)=O)C2C)=O)cc2c(ccn2C)[nH]1 N1(C(C(C)O)=O)CC23CCCC2(C1)CN(C(=O)Cc1ccc(Cl)nc1)C3 C1(C(N2CCC(N(C(c3ccnn3CC)=O)CC)C2)=O)CCC2(CCC2)C1 C1(NC(C(C)C)=O)CCOC12CCN(C(c1cc(Cl)cc([N+](=O)[O-])c1)=O)CC2 C(CCC)(C(=O)N1CCCC1CN(C(=O)CC1CCCO1)C)=CCC C(C(O)C(=O)N(CC(C)NC(c1ncoc1C1CCCO1)=O)C)=CCCC C(CN=c1nc(C(F)(F)F)cc[nH]1)=CCNC(c1nc(C)nc(O)c1)=O c1(CC(=O)Nc2c(C)nn(C)c2C(F)(F)F)cn2cccc(C)c2n1 S(=O)(=O)(c1ccsc1CBr)N.C1(C(=O)Nc2ncc(C(=O)OC)[nH]2)CCC(F)(F)C1 C#CCCCCCC(=O)N(CCC(=O)NC(CC)C(C)(C)C)C C1(c2ccccc2)(NC(C(=O)NCCCC(=O)OC)=O)CC2(CC2)C1 c1(Cn2c(-c3ccnn3C)nc(C)n2)ccc2c(C)noc2c1 c1(C(N(CCNC(c2c(C)ncn2C)=O)CC)=O)ccc2cn(C)nc2c1 c1(CC(=O)NCCOCCCNC(c2ccc(F)cn2)=O)ccccc1F N1(C(C(C)=C2CCCC2)=O)CCC(NC(=O)CCc2cn[nH]c2)C(CO)C1 N1(C(C(CC(=O)OC)C)=O)CC(N(C)C(c2ccc(F)c(C)c2)=O)C(C)(C)C1 C1(C(=O)NC2(CN(C(C3CN(C(C)=O)C3)=O)C)CC2)CCCC1C C1(NC(C2(CC=C)CC=CC2)=O)CC=C(C#CC(=O)NCCSC)C1 c1(NC(=O)OC(C)(C)C)n[nH]c2c1CN(C)CC2.C(CC1C(=O)NC12CC2)SC CC(CCC(=O)NCC=CC1CC1)NC(C1CC2(CCC2)C1)=O Cc1ccc(C(=O)NC2CC(C)N(C(c3cc(C4CCCC4)no3)=O)C2)cc1O c1(C2(C)CC2c2ccccc2)ccc(-c2noc(CS(C)(=N)=O)n2)cc1 CC1(C(=O)NCC2(C(=O)NC3CC3CO)CC2C(F)(F)F)CCCO1 N#Cc1cc(F)c(C(=O)NC2COCCC2NC(=O)CC2CCCCC2)c(F)c1 c12cc(no1)C2.N1(CCNC(C2(C(=O)OC)CC2)=O)CCC(c2nc[nH]n2)C1 Cc1cccc(C)c1C(=O)NCC1CC(CNC(=O)Cc2cnsc2)CO1 N1(C(c2c(C)ccnn2)=O)CCC(O)(C2CCN(C(=O)C3=NOC(C)C3)CC2)C1 c1(OC)c(O)cc(C(N2CCN(c3ccccn3)CC2)=O)cc1C#N N1(C(CC=C)=O)CCCCC1CC1CCN(C(c2ccccc2OC)=O)CC1 C(=O)(CC(C)(C)C#N)N1C(C)CC(NC(COCCCC(C)C)=O)C1 c1(C(=O)NC2CCN(C(c3c(Cl)cc(C)c(C)c3)=O)C2)ccc2c(c1O)CCC2 N1(C(CC2CC(NC(C)(C)C)C2)=O)CC(O)(CNC(=O)OC(C)(C)C)C1 C(=O)(CCO)N(CCC(C)C)CCCN(C)C.N(C)C C(=O)(N=c1[nH]nc(C(C)OC(C)=O)s1)NC(c1c(OC)cccc1)CC(C)C N1(C(c2c(O)ccc(N)c2)=O)CC(NC(C2(C(N)=O)CCC2)=O)C2CCCCC12 c1(C(N(CCCNC(C=CC=CCC)=O)C(C)C)=O)cnc(O)c2cccnc12 c1(CNC(C2CCN(C(=O)OC(C)(C)C)C2)=O)cc2n(n1)CCCO2 N(C1CCc2ccccc21)C(C12CN(C(C3(C#C)CCCC3)=O)C(C1)CO2)=O C12(CNC(CNC(CC)=O)=O)CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 CC1CCCCC1(C)NC(=O)C=CC1CCN(C(=O)CCn2cnc(=N)[nH]2)CC1 S(=O)(=O)(c1cc(Br)c(Br)s1)N1CCN(C(c2c(OC)nc(Br)cc2)=O)C2C1C2 n1(C2CC(C(N(CCCCC)C)=O)C2)cc(C(C2COC2)CCOC)nn1 C=CC(C)(C)CC(=O)N1CCC(C)(NC(c2cnc(SC)s2)=O)C1 N1(C(c2nnn(C)n2)=O)CCN(C(c2sccc2F)=O)CC1CS(C)(=O)=O C(=O)(CCCCC#N)N1CC(C)(OCC(=O)N(CCCCO)CC)C1 c1(CC)cnc(C(c2nnnn2C(C)C(=O)OC)NCC=C(Cl)Cl)s1 C(C)(C(=O)NC1CCCC1C(=O)N(C)Cc1ccoc1)(C(C)C)OC C(=O)(C1CC(=O)c2ccccc21)N1CC(CNC(C(C)C(C)(F)F)=O)OCCC1 CS(=O)(=O)C1CCCN(c2nnc(C3Cc4cc(Cl)ccc4O3)n2CC2CC2)C1 n1(CC#C)cccc1C(=O)N(CCC(=O)NCC1CCC(=O)O1)CC1CC1 c1(C(=O)NCC(C)(O)CNC(=O)C=CCF)ccc(O)c(Cl)n1 c1(C(=O)NCC(C)N(C(=O)Cn2cccc2)C)cnc2ccsc2c1 C1(CC(=O)N(CCCNC(c2cc(F)ccc2O)=O)CCO)CCCCC12CC2 c1(C(=O)NC(C2CCN(C(C3CCC(F)C3)=O)C2)C)cc(C(F)F)[nH]n1 C1(O)(CNC(C2CC2F)=O)CCCN(C(c2cscc2Br)=O)C1 C1(CCCC)CN(C(=O)C(F)(F)C(C)O)CCN1C(c1cocn1)=O c1(C(=O)NC(c2ccc(C)cc2)CNC(=O)C2=C(Cl)CC2)c(N)ccc(F)c1C C(N=c1[nH]c2c(c(=NCCCN3CCOCC3)[nH]1)SCC2)c1nc(C)cc(C)n1 C1(C)(C(=O)NCC2(OC)CCN(C(=O)C=C3CCN(C)C3)C2)CC2(CCC2)C1 c1(C(=O)OC)cc(Br)sc1NC(C1CSCN1C(=O)CCCOC(C)=O)=O N1(C(c2cc(OC)ncc2)=O)CCN(C(C2(C)CC2C)=O)CC(CO)C1 C1(CNC(C(=O)NCCCC(C(=O)OC)O)=O)CCS(=O)(=O)C(C)C1 Cc1cc(CC(=O)NCC2COCCN2C(=O)CCN2CCC2)n(C)n1 c1(-c2nc(CNC(N3CC(=NOC)NCC3)=O)sc2)cc2cccc(OC)c2o1 c1(C(N2C(CC(=O)NCCCN(OC)C)CC2)=O)cnc(C)nc1C CC1(C)CC(C(=O)N2CCCC2CNC(c2nc(Cl)ccc2F)=O)=NO1 C1(C(C)(C)NC(C(CC)OCC)=O)CCCCN1C(c1csc(CC)n1)=O C1(C(=O)Nc2cccc(Cl)c2)(CC)CCCN(C(=O)Cc2ccc(O)cn2)C1 C1(CN(C)CCOCCNC(=O)CCCCc2cccs2)CCCC(F)(F)C1 c1(C(N(C(C)CCNC(=O)CCOc2cccnc2)C)=O)ccc2cnoc2c1 c1(C(=O)NC2C(NC(CC(C)SC)=O)CCC2)coc2c1COC2 c1(C(=O)NCC23C(CN(C(c4ccn(CC#N)n4)=O)C2)C3)ccc2n[nH]cc2c1 N1(C(CC(C)c2cnn(C)c2)=O)CCC(CNC(C2(CCO)CC2)=O)C12CCC2 C(=O)(C#CC1(C)COC1)N(CCCNC(c1c(C2CC2)ccc(C)c1)=O)C(C)C C1(NC(C2C(C=C)OCC2)=O)CCN(C(c2oc(C)nc2C)=O)C12CCC2 c1(C2C(C(=O)NCCCCNC(c3ccnnc3O)=O)C2)ccc(F)cc1F c1(NC(C(C)C)C)ccc(S(=O)(=O)NCC(C)CCO)cc1F N1(C(CP(C)(C)=O)=O)CC(CNC(C2CCC3(CCC3)C2)=O)CC1(C)C C1(CNC(CSSC)=O)CC2(CCN(C(c3cc(C)cc(Cl)c3)=O)CC2)CO1 C12(C(N3CC4CC(NC(CS(CC)(=O)=O)=O)C4C3)=O)C3C(=O)C4C5CC(C14)C2C35 c1(OC(c2nnc(N(C)C)n2CCC#N)C)cc(Br)cc(F)c1F Cc1nscc1CC(=O)NC(C)CN(C(=O)CCc1cncs1)C CCCCCCCC(=O)N1CCN(Cc2ccc(Br)s2)CC1CC C1(C)(C(=O)NC(CNC(C=Cc2cncc(C)c2)=O)C2CC2)CC2CCC(C1)S2 C(=O)(C(C)(C)Cc1ccccc1)NCC(=O)N(C)CC c1(CC)cc(C)ccc1C(=O)N(CCNC(=O)Cc1ccc(CO)cc1)CC c1(C(N2CC3(C(NC(CC(C(C)C)O)=O)CCS3)C2)=O)cc2nn[nH]c2cc1F Cc1cncnc1C(N1CCCC(CCNC(=O)CCc2csc(=N)[nH]2)C1)=O N1(C(C2C(C)(C)CCCC2)=O)CCN(C(c2ccc3cnoc3c2)=O)CC(O)C1 c1(CC)ccc(C(=O)NCC2CN(C(=O)C(C)n3cnnn3)CCO2)cc1Cl c1(OCC)ccc(C(=O)NCCN(C(=O)CC2CCSCC2)CC)nc1 C1(OC)CCn2cc(C(=O)N(C(C)CN(C(=O)C(F)=C3CCCC3)C)C)nc2C1 N1(NC(C(C)OCCOCC)=O)CCC(NC(=O)Cn2nnc(=O)[nH]2)CC1 C1(NC(c2cn(CCC)nc2)=O)CC2CN(C(=O)CC3CCCN3C)CC12 c1(CN2C(CC(=O)OC)CCC2)no[nH]c1=NC(=O)Nc1cc(B(O)O)co1 C(=O)(C1=C(C)OCC1)N1C(CN(CCCC=C)C)COCC1 N1(C(c2c(C)cncc2)=O)CCCN(C(c2ccccc2S(C)=O)=O)CC1C N1(C(CCN(C(=O)OCC)C)=O)CCC(C(=O)NC(C)CNC(=O)NC)CC1 C1(CC(=O)NCC2(O)CN(C(COC3(C)CCCC3)=O)C2)CCS(=O)(=O)C1 C(=O)(C1=NNC(=O)CC1)NCC(C1(O)CCN(C(C2=C(C)CC2)=O)C1)C Cc1ncnc(C(=O)NC(C)(CNC(=O)C(O)C2CCCC2)C(C)C)c1C c1(C(N2CC(NC(c3ccc(C=C)cc3)=O)C(F)C2)=O)c(F)ccc2ccoc12 c1(NC(C2CCN(CC3(C(=O)NC)CC(=C)C3)C2)=O)cc(C)c(C)c(C)c1 N1(C(C2CN(C(=O)C3CC3)C2)=O)CCN(C(C2CNC(=O)C2)=O)C(CO)C1 C1(C#N)(C(=O)NC(C)CN(C(=O)Cc2cnccn2)C)CC1(C)C C1(CNC(C(CC)n2cccn2)=O)CN(C(c2oc(CO)nc2C)=O)CC12CC2 c1(C(=O)OC)cnc[nH]c1=NCC1CCCC12CN(C(=O)C1=NNC(=O)C1)C2 N1(C(CC(CCC)C)=O)CC2CCC1C(CNC(=O)C(C)OCC1CC1)C2 c1(C(N2CCC(NC(C)=O)CC2)=O)cn(C)c(=O)n(C)c1=O.N1(CC)CCCC1 c1(NC(C2C(NC(c3cc(OC)cc(I)c3)=O)C2)=O)cc(Cl)c(Br)cc1[N+](=O)[O-] c1(CC(=O)NC23CC(CNC(CC(C)F)=O)(C2)C3)cc(Br)ccc1Br C(CC1CC1)(C(=O)NCCSC)OC.c1(C(=O)O)cnco1.C12CC1C(=O)NC2C Cc1ccc2c(c1)ncn2CC(=O)NCCC(C)NC(c1cc(O)ccc1F)=O c1(NC(C(C)=CC(C)(C)C)=O)cccc(NC(c2sc(C)nc2CC(C)C)=O)c1 Cc1cccc(C)c1NC(C1CC12CCN(C(c1cc(F)nc(F)c1)=O)C2)=O c1(C(N2CC(C)N(C(=O)CSC(F)F)CC2)=O)cc2cccnc2cc1F N1(C(CONC(Cc2ccn(CC)n2)=O)=O)CCC(O)(C#CBr)CC1 Clc1ccc(C2(C3CCCOCC3)CC2)cc1.c12nc(no1)CCNC1CC21 C(CCCCC(=O)NC1CC2CCC1(NC(c1cc(CCCO)on1)=O)C2)OC c1(C(=O)NCC(CC)NC(C2CC=CCC2)=O)nccc(OC)c1F N1(C(c2nc(C)oc2)=O)CC(NC(c2cc(Cl)c(Cl)s2)=O)C(O)C1 O=C1CN(Cc2nc(Cn3nccn3)n(-c3ccccc3)n2)C(=O)CN1 N1(C(c2cccc(NC)n2)=O)CC2CCCC2(NC(c2ccc(C3CC3)o2)=O)C1 N1(C(=O)N=c2[nH]nc(CC3CCCC3)s2)CCOc2c(Br)cccc2C1 c1(N(C(=O)NC(C)CCC2CCCCC2)CC#N)cncc(Cl)n1 CCCCC(CNC(=O)C(CC)Oc1cccc(Cl)c1)NC(C1CC1C(N)=O)=O c1(-c2cn(CCCC(N3CCC(C)CC3)=O)nn2)c[nH]c2ncccc12 c1(C(C(=O)C(=O)CC2(OC)CCC2)=O)ccc(OC)c(O)c1.CCCNCCC(=O)OC N1(C(CC(=O)N(C)CCN(C(CC(C)C)=O)C)=O)CCOC(c2ccco2)C1 C(=O)(N1CCOC1=S)N1CCCCC1OC(CC)C c1(C(=O)NC2(C(C)NC(C3NC(=O)CC3C)=O)CC2)ccc(C#CC2CC2)cc1 c1(C(=O)NCC#CCNC(COC(C)=O)=O)ccc(-n2ccnc2)c([N+](=O)[O-])c1 N1(C(C(C)=CC)=O)CCCCC(NC(=O)OC)C1.C1(=O)CC(C)N1C C(=O)(CCCC(F)(F)F)N1CC(CCO)(NC(C(CC=CCC)C)=O)C1 Cc1cc(CNC(C2(CF)CCN(C(=O)CNC(=O)CN(C)C)C2)=O)ccc1F c1(OC)cccc(CC(=O)NC(C)CCCNC(c2ccnc(Cl)c2N)=O)c1Cl c1(C(N2CCC(NC(c3c(OC)nccc3)=O)C(C)C2)=O)cc(F)c(C)cc1F CCC(CC)CC(=O)NC(C1CN(C(=O)CN2CSCCSC2)C1)C C1(CNC(C(C)N2CCCC2)=O)CCC(C(=O)NCc2noc(N(C)C)n2)O1 N=c1nc(N2CCc3c(F)cccc3C2)[nH]c(=NC2CNC(=O)C2)[nH]1 c1(CC(=O)NC(CC)CNC(=O)C(C)C2CCC2)cc2ccccc2nc1O NC(=O)C1=NOC(CNC(C2CCN(C(=O)C=Cc3ccsc3)CC2)=O)C1 c1(CNCC2(OCC)CCOC2)c(C)cnn1C c1(C(N(CCN(C(=O)C(F)(F)c2cccnc2)C)C)=O)ccnc2ncccc12 CC1(C(=O)NC(c2ccc(Cl)cc2O)=O)CCN(Cc2c[nH]cc2Br)CC1 Cc1nn2cc(C(N3CCC(NC(=O)CSC(F)(F)F)CC3)=O)nc2s1 C1(CNC(c2ncc(OCC)nc2)=O)CN(C(=O)CNC(N)=O)CC1(C)C CC1CN(C(=O)CC2CSC2)CC(C)N(C(=O)C=CSc2nc[nH]n2)C1 N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)C(NC(c2cccnc2O)=O)C1 c1(C(N2CC(NC(c3ccc(C)c(C)c3)=O)C(O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(N2CCCCC(SC)C2)C(=O)NCCCOC)cc(Cl)c(C)cc1Br C(=O)(C1CCC2(CCC2)C1)N1CCN(C(C=Cc2ccn(C)c2)=O)CC1 Cc1noc(CC(=O)NCc2nc(C(=O)NCCCOC3CCCC3)co2)n1 C(=O)(C(C)C(F)(F)F)NCC(C)OC.C(=O)(CCOCC)N(C(CC)C)C C(c1ccc(F)cc1)=CC(=O)N(CC(C)CNC(c1coc(CC2CC2)n1)=O)C C1(CC(=O)N(CCCC(=O)N2CC(NC(C)=O)C2)C2CC2)CCCOCC1 c1(OCC)ncccc1C(=O)N(C)CC1(O)CN(C(C2CC2(C)C(C)C)=O)C1 C1(NC(=O)C=CC)CCCCC1.c1(C(=O)NCC(CO)NC(=O)CS)ccco1 c1(CC(=O)NC(C)CCCCNC(c2cnc(S)[nH]2)=O)c[nH]c2cccc(F)c12 c1(C(c2n(CCCC)nnn2)NCC(=O)OCc2ccsc2)ncc(Cl)cc1Cl CCC(CC)CC(=O)N(C)CCN(C(=O)CC1OCCOC1(C)C)C c1(C(=O)NC2CC3(CC(NC(C(C)C4CCOC4)=O)C3)C2)ccn2ncccc12 N1(C(C2(CC)CCC2)=O)CCC(CNC(C2CCC(=O)N2)=O)CC1 C1(N(CC(C)C)C(c2cnco2)=O)CCN(C(C2CCC(O)CC2)=O)CC1 C(=O)(C(CC(C)C)CC(C)C)NC1C(OC)CN(C(c2ncccc2F)=O)C1 c1(C(N2C(C(N3CCCC3C(F)(F)F)=O)COCC2)=O)ccc(I)cc1[N+](=O)[O-] C1(N(CC(c2ccccn2)O)C(c2c(C)onc2)=O)C2CCC1CNC2 N1(C(c2onc(C)n2)=O)CCC2(CCCN(C(=O)CCC(C)N(C)C)C2)C1 c1(C(=O)NC(c2ccnn2C)C(=O)NC2C(CCC)CCC2)nc(C)ccc1C C1(CNC(c2cccc(Br)c2)=O)CC(F)CN1C(=O)Cn1cnnc1O C1(NC(C2(NC(c3c(CC)c[nH]n3)=O)CC2(C)C)=O)CCCC(C(N)=O)C1 C(=O)(CCC1=CCCCC1)NCC12N(C(=O)COC3CCCC3)CC(CC)(C1)C2 C1(CCNC(c2ccoc2)=O)COCCN1C(=O)C1=CCSC1 N1(C(C2N(C(=O)OCC)CSC2)=O)CCC(C2(NC(c3coc(Br)c3)=O)CC2)C1 c1(C(=O)NC(CC)CN(C)C(C2CC23CCC3)=O)cc(C)n(C(C)(C)C)n1 N1(C(CC)=O)CCCN(C(C(=O)NCC2CCCO2)C(C2CCCC2)C2CC2)CC1 C12(NC(C=CCOC)=O)CC(C)(C1)OC21CN(C(c2nn(C)cc2SC)=O)C1 C1(C(=O)NC(C(=O)NCCc2n(C)ncn2)Cc2cn[nH]c2)Cc2nccn2C1 c1(C(C)F)cccc(NC(C2(c3cnn(C)c3)CCCO2)=O)c1 C(=O)(C(=O)CCCC)N1C(C(=O)NC(C=C)C)COCC1 N1(CCc2cn(CCS)nn2)CCCN(C(=O)C(C)c2ccsn2)CC1.CC(=O)O C(C(C)(O)C(=O)N1CCN(CC(=O)NCCC2CC(C)=NO2)CC1)OC Cc1ccc(-c2nc(CCC3CCCN3C)n(Cc3ccsc3)n2)cc1Br C1(NC(CC=C)=O)CCC(C)N(C(c2cn(-c3nonc3CC)cn2)=O)C1 Cc1sc(C(=O)NCCCCC(C)NC(=O)C=CBr)cc1Br Nc1cc(C(=O)NC2CC2CNC(c2cnn(C3CC3)c2)=O)ccc1Br c1(CN(C(=O)NCc2c(OC)nccc2)C)cccc(C)c1F Cc1ncn(C)c(=O)c1C(=O)NCC(C)N(C(=O)C(c1ccc(F)c(F)c1)O)C C1(CC=C)(NC(=O)C(F)(F)c2ccccc2)CCN(C(=O)CC(=O)N(C)C)C1 CC1CC(NC(c2nc(Cl)c(Cl)s2)=O)CN1C(=O)Cc1cccnc1 CC(C)CC(O)C(=O)NC1(CCCNC(=O)COC(=O)N(C)C)CC1 CC1(C)C(C(N2CCN(C3CCN(C(c4sccc4Cl)=O)C3)CC2)=O)C1(C)C Cc1ccc(NC(c2sccc2NCc2ccc(O)c(Cl)c2)=O)c(C#N)c1 CC1(C)COCCC1NC(=NCCc1cccnc1)NC(CF)CF C1(=O)C(C)(C)C(=O)N2CCCC(C2)N1.S(=O)(=O)(CC(F)(F)F)N(CC(=O)O)CC CC(C)CC(C)(CNC(C1(C)C(C)(C)C1(C)C)=O)NC(C1CCCOCC1)=O C1(C(=O)NC2CC3(CN(C(c4c(CCC)nns4)=O)C3)C2)CC(=O)N(C)C(=O)N1 N1(C(C2(C)C=CCCC2)=O)CCCC(CC(=O)Nc2cncc(Cl)c2)CC1 CP(C)(=O)CN1CCOC(C(=O)NC2CN(C(=O)Cc3cnccn3)C2)C1 CP(C)(=O)C(CCNC(=O)CNC(c1ccc(Cl)cc1F)=O)c1ccccc1 CN1CC(F)CC1C(=O)NCCN(C(=O)C(O)Cn1cncn1)C1CCCC1 Cc1cccc(-c2ccnc(CNCc3c[nH]c4cccnc34)c2)c1[N+](=O)[O-] C=CCCC(CC(C)C)C(=O)NC1CC(C)CN(C(c2nn[nH]c2Cl)=O)C1 N1(C(C(C=C)O)=O)CCCC1(c1cn(CC2C(C)C2(F)F)nn1)C(F)(F)F CCCC(CC)CCC(=O)N1CC(CC(N(C)CP(C)(C)=O)=O)CC1C CN1CC(F)CC1C(=O)NCCNC(=O)C(=O)Nc1ncc[nH]1 CC#CCCCC(=O)N1CCC(NC(=O)C2CC2)C1C N1(C(=O)NC(C)C)CCC(C(=O)NC(C)CN(C(=O)CS(C)(=O)=O)C(C)C)CC1 C1(NC(c2ncn(C)n2)=O)CC(CNC(c2cnc[nH]2)=O)C1(C)C C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(c1cccc2nc(C(F)F)[nH]c12)=O c1(C(=O)NCC2CCCC(NC(c3cccc(F)c3)=O)C2)cc(O)ccc1Cl n1(CC)nncc1C(C(=O)NCCCSC)N(C)Cc1scnc1C Cc1cncc(C(=O)NC(C2CC(NC(c3cnn(C)c3)=O)C2)C)n1 N1(C(c2cnc(C)[nH]2)=O)CCN(CC(C)(C)NC(=O)C2=CCCC2)CC1 N1(C(C(C)S)=O)CCC(O)C(C(=O)NC2CNC(=O)C2(C)C)C1 c1(C(N2C(CC)C(C(=O)N(CC(F)(F)CO)C)CC2)=O)cccc2[nH]ncc12 C(c1cc2ccccc2o1)=CC(=O)NC12CC(NC(=O)CC3COC(=O)N3)(C1)C2 C(CCC)(C(O)C(=O)N1CCC(OCC)C1C)NC(C(C)=CCC)=O N1(CC)N=C(C(=O)N2CC3CC3(CNC(c3nncn3CC)=O)C2)CCC1=O N1(C(C(C(=O)OC)C)=O)CCCC(C2CC2NC(c2cc3n(n2)CCOC3)=O)C1 C(CCCC(=O)NCCCCCCNC(C1CC1(C)C(C)C)=O)NC(C)=O C1(CNC(c2c(CCC)nco2)=O)CC2(CCN(C(=O)C3=CCCO3)C2)CO1 N1(C(c2c[nH]c(=NC)o2)=O)CCCC12CCN(C(C1CC3CC(O)C(C1)C3)=O)C2 C1(CC)CN(C(=O)C=CC2CCC2)CCN1C(c1sc(Br)cc1F)=O c1(C(=O)NCCC2CN(C(C3CCOC3)=O)CCO2)cc(O)ccc1Br C1(C(=O)NCC(CNC(C(C)CCn2cccn2)=O)(F)F)CCc2c[nH]nc2C1 c1(NC(c2cc(CC3CC3)on2)=O)cc(CO)c(Cl)c(Cl)c1 C1(C(C)(C)NC(C(C)=CC2CC2)=O)CCN(C(C23CCCC2CC3)=O)CC1 c1(C(=O)NC(C2CCN(C(C3C(=C)C3)=O)CC2)C)cc2c(nn1)CCCC2 C(=O)(C(C)CC(C)C(C)=O)NC(C(=O)Nc1cccc(C#C)c1)(C)C C1(CC)CN(C(=O)C(O)C2CCC2)CCN1C(C1CCC2(CC1)CC2)=O C1(C(N(CC(C)NC(=O)Cc2ccccc2F)C)=O)CCn2cncc2C1 N1(Cc2nnc(-c3cccc(C)c3)o2)CCc2c(cnn2C)C1 c1(C(=O)NC(C(C(C)C)NC(=O)Cc2cnc[nH]2)C)cccc(C(F)F)c1F C(C(C)(CC)C(=O)NCc1[nH]nnc1C)NC(C(CC)C#N)=O CC(O)C(F)(F)C(=O)NCC1CC1NC(C1(c2ccc(F)c(F)c2)CCCC1)=O C(=O)(C(C(C)(C)C)OC)NCCN(C(C1CN(CC(F)(F)F)C1)=O)CC C1(C(=O)NCC2CC(F)(F)C2)CCCN(C(=O)Nc2ncccn2)C1 c1(C(N2CC(CNC(C=C3C(C)(C)CCCC3)=O)C2)=O)ccc2nnc(S)n2c1 C#CCCCC(=O)N1CCCC1CCNC(c1cnc(C2CC2)nc1)=O C1(C2N(C(C3(CF)CCC3)=O)CC2)CCCCO1 N1(C(CS(CC)(=O)=O)=O)C(CNC(=O)Cc2ccno2)CC2CCCCC12 c1(C(=O)NCC2(OC)CCCN(C(c3occc3CN)=O)C2)ccc(C#N)cn1 C1(C(=O)NCc2nccc(C)c2)CCC2CCC1N2C(c1[nH]ccc1C1CC1)=O C(=O)(C1=CCN(CC)C1)N(C(C(c1ccccc1)CC)=O)Cc1ccc(Cl)cc1 c1(C(=O)OC)ccc(NC(C2CN(C(=O)C(C)(F)F)CCS2)=O)cc1OC c1(CC(=O)NCCCN(C(C2N(CC)CCOC2)=O)C)ccc(OCC)cc1F C1(COC)CN(C(=O)CSc2nncn2C)CCN1C(c1ccn(CC#N)n1)=O c1(C(=O)NCCC2(O)CCN(C(CC=C)=O)C2)cc(Cl)ccc1OC(F)F C1(C(N2CCC(C)(N(C)CC)C2)=O)CN(C(c2ccccn2)=O)CCC1(C)C c1(C(=O)NC2CC2CNC(c2[nH]ccc2-c2ccccc2)=O)cccnc1Cl c1(NCC=C(C)C)nc2ccccc2nc1NC1CCC(C)(C)CC1 Cc1c(F)ccc(C(N2CCC(C(=O)Nc3cc(Br)nc(Br)c3)C(O)C2)=O)c1Cl Cc1cc(CNC(=O)CCOCCN(C(=O)CCCN(C)C)C)cnc1Cl N1(CCC(=O)N(CCC)CCNC(C2(CF)CCC2)=O)CCNC(=O)C1 C1(C)(CNC(CC2CCN(C(C(c3cncnc3)C)=O)C2)=O)CCN(C)C1 C1(NC(c2c[nH]nc2-c2cccs2)=O)CCSC12CN(C(=O)C=CC1CC1)C2 C1(F)(CNC(C(C)Cc2cnco2)=O)CCN(C(C2(C(F)(F)F)CCO2)=O)C1 N1(C(c2ccc(CC)s2)=O)CCC(C(=O)NCC(C)Cc2cn[nH]c2)C1C c1(C(N(CC(=O)NC(CO)C2CCC2)Cc2ccccc2)OC)ccncc1Cl c1(C(=O)NC2(C)CCN(C(c3cnn(C)c3N)=O)C2)cccc([N+](=O)[O-])c1 C1(C(=O)NCCOC2CCN(C(c3cn(CCOC)nc3)=O)C2)CC(=O)N(C)C1 N1(C(c2c(C)sc(O)n2)=O)CC2CC1CN2C(=O)CC1CCCNC(=O)C1 c1(C(=O)NC(C)CNC(=O)C=Cc2cocn2)ccc([N+](=O)[O-])c(N(C)C)c1 c1(C(=O)NC2(CC)CCN(C(=O)CCOC)CC2)ccn2ncccc12 Cc1cccc(CC(N2CC(OCCNC(=O)Cc3ccccc3O)C2)=O)c1Cl C12(NC(C=CCN(C)CC)=O)CC(C(N3CCC(CN(C)C)C3)=O)(C1)C2 C1(NC(=O)CCc2nc[nH]n2)CN(C(c2cc(Cl)n[nH]2)=O)CC1C1CC1 CS(=O)(=O)C1(C(=O)NCC=CCNC(c2cnn(C3CCCC3)c2)=O)CCCC1 c1(C(=O)NC2CCCCN(C(C(C)=C3CCC3)=O)C2)c(C)nc(C2CC2)nc1O C(CN=c1[nH]c(N2CCC(N3CCC3)C2)nc2ccccc12)C1S(=O)(=O)CCC1 C(CO)(CO)(C(=O)O)NC(C1CCN(Cc2ccccc2)C1=O)=O C1(NC(=O)CCF)CCOCC1NC(c1nccnc1C(N)=O)=O C#CC1(C(=O)NC2CC(NC(c3ccccc3C(=O)OC(C)(C)C)=O)C2)CCCC1 c1(NC2C(C(=O)Nc3c(I)ccc(C)n3)C2)ccn2ncc(Br)c2n1 Cc1c(C=CC(=O)NC2CC3CCC2(NC(c2cnsc2)=O)C3)cnn1C CC(O)C(F)(F)C(=O)NC1COCC1CNC(=O)Cn1cnc(=N)[nH]1 c1(C(N2CCCC(C(CNC(CC(=C)C)=O)(C)O)C2)=O)ncc(N)cc1Cl n1(CC(=O)NC2CN(C(Cc3cnc(C)o3)=O)CC2O)ccc([N+](=O)[O-])n1 c1(C2(C)CC2)ccccc1C(=O)NCCCNC(=O)CC1CCCC(=O)O1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(CNC(C2CC2F)=O)OC2CCCC12 CCC(CC)C(C(=O)N1CC(C(N2CCC(CC3CC3)C2)=O)CCC1(C)C)OC C(=O)(C1=C(C)OCCS1)N1CC(CC(=O)NCc2cc(C)cc(C)n2)(OC)C1 C(C(C)(C)C#CC(=O)NC(CO)CCO)NC(C(CCOC)C)=O C1(c2ccccc2)(C(=O)NC2CN(C(=O)C=CCF)C2)CCCO1 Cc1ccc(CSCC(=O)NC2CN(C(=O)C(C)(C)C)CCO2)cc1 c1(COCC)n[nH]c(=NC2CC(CCNC(=O)CN=S(C)(C)=O)C2)s1 N1(C(C(CN=[N+]=[N-])NC(C=C(C)C)=O)=O)CCOCC2(CCC2)C1 CCCC(CCC)C(=O)NC1CCCCCC1NC(C1CCCCN1N=O)=O C1(NC(C(CNC(CCc2cc(C)[nH]n2)=O)O)=O)CN(C)C(C)(C)C1 c1(C(N(C)CC2N(C(CCCC#CC)=O)CCOC2)=O)c([N+](=O)[O-])cnn1C Cc1cc(C)n(CCNC2(c3nnnn3C3CC3)COC(CO)C2)n1 c1(N(C(C2CCC(F)CC2)C(=O)NC(CC)(C)C)C)ccccc1Cl CN=c1nc(N2CCC(c3cc(O)n[nH]3)C2)[nH]c(=NC(C)Cn2cncn2)[nH]1 C1(n2c(-c3cnn4cccc(Cl)c34)nc(C(C)(C)C)n2)CCc2ccccc2C1 C1(NC(C2CC(OC)C2)=O)CN(C(=O)Cc2cccnc2F)CC1(C)C c1(C(N2CCCC(CNC(C3C4CCCC34)=O)CC2)=O)cnc2ncccn12 N1(C(CCSCCC)=O)CCCC(O)(CNC(C2CC(CCC)C2)=O)C1 Cc1cccc(F)c1CC(=O)NCCC1(CNC(=O)C=CCN2CCCC2)CC1 N1(C(C2C(OC)C2)=O)CCC(C)(CNC(c2ccccc2OCC(N)=O)=O)CC1 C(CC(C(=O)N1CCC(OCCOC)C1)NC(c1cc(O)nn1C)=O)OCC C(C(C)(C(=O)NCC(C1CCN(C(=O)COC2CCOC2)CC1)O)OC)OC Cc1csc(=O)n1CCC(=O)NC1CC1NC(=O)COc1cnn(C)c1 C12(NC(CC=CC)=O)CCC(CNC(C3CC34CC4(F)F)=O)(CC1)OC2 CCCC(O)C(=O)N1CC(NC(c2cc(-n3cccc3)ccn2)=O)C(SC)C1 N1(C(c2occ(C)c2C)=O)CC2CC(C1)CN(C(C1COCCC1C)=O)C2 c1(CC(=O)N(C)CCNC(=O)CC2CC2(Cl)Cl)cc(F)cc(Br)c1 CC1(C)OCCC1C(N1CCC(OCCNC(=O)CNC(c2ccsc2)=O)C1)=O c1(CC(=O)NCC2CN(C(c3c(C)cco3)=O)C(C)(C)C2)ccc([N+](=O)[O-])cc1 C1(CNC(c2n[nH]cc2Cl)=O)CCCCN1C(c1coc(C2CCC2)n1)=O C1(C(N2CCN(C(CNC(C(F)=CC)=O)C)CC2)=O)Cc2nc(C)cn2C1 N1(C(Cc2cc(C)sc2)=O)CCOCC1CNC(c1nccnc1C)=O Cc1ncc2c(n1)CCC(NC(=O)CSc1ccccc1O)C2 c1(C(N(CC(C)CNC(=O)C2=CCS(=O)(=O)C2)C)=O)cnn2c1CN(C)CC2 CC(C)(C)C(CNC(C1CCCC12CCC2)=O)C(=O)N1CCC(F)(F)C1 N1(C(C2(c3ccc(C)nc3)CC2)=O)C(C)CC2CN(C(C3CCCN3C)=O)CC12 c1(NC)nc(C)ccc1C(=O)NC1CC(NC(=O)CCCC2CCCC2)C(O)C1 N1(C(CC(C(=C)C)OC)=O)CCC(C)(C)CC1C(N1CCCC1CSC)=O N1(C(c2cc(OC)ncn2)=O)CCC2CC2(NC(C2(F)CC2)=O)CC1 C1(CCNC(C=CCOC)=O)CCN(C(c2cccn2C)=O)C1 C1(NC(c2c(CC)scc2)=O)CC2CC(NC(=O)C=Cc3sccc3C)CC12 N1(C(C2(CC#C)CCOC2)=O)CCC2(C=C(C(=O)N3CC(O)CC3C3CC3)C2)C1 C1(NC(=O)CC2CCCCC2(F)F)CC1C1CCCN(C(=O)C=CCO)C1 Cc1cc(Cl)c(C(=O)N(C2CC(N(C)C(C3CCC4CC4CC3)=O)C2)CC)cc1F Cc1cnc(NC2CCN(C(=O)CCCN3CCCCC3)CC2)nc1C N1(C(C(CC=C)c2ccccc2)=O)CCCC(O)(c2cn(C(C)CC)nn2)C1 C=C(Br)CC(C)(C)C(=O)N1CCC2(CC1)CC2C(=O)NCCOC Cc1[nH]nc(C(N2CC3CC(NC(C4CCOCC4)=O)CC3C2)=O)c1[N+](=O)[O-] C1(N(C(c2ccncc2)CCC)C(c2ccco2)=O)CCNCCC1C c1(OC)cc(NC(c2ccc(-c3cccc(N)c3C)cc2)=O)c(N)cc1F c1(C(N2C(CN(C(C)C)Cc3cc(C)on3)CCC2)=O)cccc(C(N)=O)c1F C1(CCC)CCCCN1C(=O)C(O)CNC(=O)C(c1ccn(C)c1)C Cc1ncc(CN2CC(CNc3nc(C(=O)O)c(C)s3)CC(C)C2)c(O)n1 C1(CNC(=O)Cc2cc[nH]c2)(NC(C2CC(N3CCOCC3)C2)=O)CCCC1 Cc1c(C(C)C)n[nH]c1C(=O)NCC(CC(C)C)NC(=O)CN1CCC(O)CC1 C1(C(N2CC(CCOC)N(C(C3CC4CC3C4)=O)CC2)=O)CC1C1CCCCC1 C1(NC(C2(CC(C)=O)CC2)=O)CCOCC1C=O.c1(C2CCC2)ccn(C)n1 c1(C(=O)NCC2N(C(C(CCC)C)=O)CC2)ccc(OCC)cc1.c1(O)cccc(C)c1 c1(C(=O)NCC2CC(NC(C(CCSC)O)=O)C2)cnn2c(O)cc(C)nc12 c1(-c2ccc(C(=O)NC3(CNC(COC(CC)C)=O)CC3)o2)ncccc1Cl N1(C(C(=O)NC2CN(C)C2)=O)CCC2CN(C(=O)OCCOC(C)(C)C)CC2CC1 C1(CNC(=O)C=CC2CCC2)C2CC1N(C(=O)CCC1CC1(F)F)C2 NC1CC2(CCC(C(=O)NCC3(Sc4ccccc4)CC3)CC2)C1 C(CCCCCCO)SCC(=O)NC(C1CCC(NC(=O)C(C)(C)C)C1)C CC(=O)NCC(NC(=O)C=CC(=O)N)CC.C(C)(C)(C)OCC1CC1 C(CCC(CO)NC(c1ccc(C(OC)OC)s1)=O)NC(c1c(CC)scn1)=O c1(C(N2CC(OCC)C(CNC(=O)COC)C2)=O)cccc(Br)c1F C(C(C)(C(F)F)NC(=O)CC1CCCC12CC2)OC c1(C(C)C)ccc(CC(=O)NCC(Cc2ccccc2)N(C(=O)C(N)=O)C)cc1 c1(CC)cc(N)ccc1C(N1CC(O)(CO)C1)=O.C12(CCCCC1)CC(=O)N2C O=C(CCC=CBr)NCC1(CNC(=O)C=Cc2cocn2)CCCC1 C1(NC(C(CNC(COCC(=O)OCC)=O)OC)=O)CC2(CNC(=O)O2)C1 C1(NC(c2ccc(-c3ccc(Br)cc3)s2)=O)CCn2ccnc2C1 C1(CC)(NC(C2OCCC2C)=O)CN(C(=O)CNC=O)C1 C1(C(=O)OC)CCC(C(=O)N(CCCSC)CCNC(=O)C=Cc2ncco2)C1 c1(C(N2C3C(NC(=O)CC4CCNC4=O)C(CC3)C2)=O)cc(F)c(F)cc1F c1(C(N2CCC(C)(C(N3CCC(CC)C3C(C)C)=O)C2)=O)cc(C#N)[nH]c1C N12CCOC(C1)C2.c1(C(=O)OC(C)(C)C)nc(CCc2ccccc2)cs1 c1(CCCC(N2CCCC(C(=O)O)(CC)C2)=O)c[nH]c2ccccc12 N1(C(CC2C(CC)C2)=O)CCC(CO)(NC(=O)CSc2nnnn2C)C1 Cc1cccc2nc(CNC(c3ccc(CSC4CC4)nc3)=O)cn12 c1(C(N2CC(N(C)C(c3scnc3Cl)=O)C2)=O)ccc2c(c1)C(=O)CCO2 C1(NC(C(C2CC(F)(F)C2)OC)=O)CC(Nc2cncc(Cl)n2)C1(C)C C12(C(=O)OC)CCCC1CCN2C(=O)Cn1cc(C2(N(C)C)CC2)nn1 c1(C(N(CC(C)(C)CNC(=O)CC2CC23CC3)C)=O)cnc2c(c1)OCC(=O)N2 CCCC(CC(=O)NCC(C1CCC1)O)NC(=O)Cc1ccn(C)c1 c1(C(N2C(C)C(NC(=O)CCc3ccc(F)cc3)CC2)=O)ccc2nn[nH]c2c1 c1(C(=O)OC)cc(NCC2CCSC2(C)C)nn2c(Br)cnc12 c1(C(N2CCCN(C(C(C=C=C)C)=O)CC2C)=O)cn(C)c(=O)c2ccccc12 C(CCC(C)(C)NC(=O)CC1CCN(C(=O)CN2CCCC2C)CC1)OC c1(C(=O)NC(CNC(C(C(C)C)NC(N)=O)=O)C)occ2c1CCC2 C1(C(N(C2CCCCC2)CC)=O)CC(O)CN1C(c1scnc1C(F)(F)F)=O CC(=O)C(C)CC(C)C(=O)NCC(C)(C)NC(=O)C1=CC(C)(C)C1 CC1(CC(=O)NCC2CCCC2NC(=O)CSCc2cscn2)CC1(F)F N1(C(c2cc(OC)nc(Cl)c2)=O)CCCCC(N=c2cc[nH]cc2[N+](=O)[O-])C1 N1(C(=O)COC(F)(F)F)CCC2C(C1)CN2C(=O)CC1CCSCC1 CC1=C(C(=O)NCC2CCCCN(C(c3nc(=N)cc[nH]3)=O)C2)C(C)(C)CCC1 N1(C(CC2CCN(C(CNC(N)=O)=O)CC2)=O)CCC(O)C(F)CC1 n1(CC)nc(C(N2CCC(CO)C(NC(=O)CCc3ccoc3)C2)=O)ccc1=O C1(NC(C(CC)=CC)=O)(CO)CCN(C(c2cc(Br)cn2C)=O)C1 N1(C(CCCCC)=O)CCCC(C)C1CNC(C1CC(N2CCOCC2)C1)=O S(=O)(=O)(c1ccc(Br)cc1NCCc1ccccc1Br)N1CC(C)(C)C(CO)C1 C1(CNC(C2CCC(NCc3cc(C(=O)OC)[nH]c3)C2)=O)CC2CCC1C2 C1(NC(C2ON=C(CC)C2)=O)CC2(NC(=O)CNC(C3CCCC3)=O)COC1C2 Cc1c(C(=O)NCC2(O)CN(C(=O)C=Cc3ccn(C)c3)C2)cnn1CC(F)F C1(NC(C=CC(C)NC(=O)CC2CSCCO2)=O)CC2(C1)CC(C#N)C2 c1(NC(=O)NCc2onc(-c3ccc(OC)cc3)n2)c(F)cc(C)cc1Cl C(C)(CC(C)NC(C1CCOC1)=O)NC(C1C(=C)C1)=O C1(OCC)CN(C(=O)CCC(CC)OC)CC1NC(c1cc(C2CC2)on1)=O c1(C(C)NC(c2nnnn2CCCC2CC2)(C)CC2CCCC2)ccnc(F)c1 c1(C(C(N2CC(NC(=O)Cn3nccn3)C2)=O)O)cccc(F)c1 Cc1nc(O)[nH]c1C(=O)NCC1(CO)CCN(C(C2(C)CC=CCC2)=O)C1 C1(CC#C)(C(N2CCCC(NC(=O)CCOCC(=C)C)C2)=O)CCOCC1 C12(COC)CC(NC(=O)Cc3ccco3)(CN1C(c1cc(C)ncc1Cl)=O)C2 c1(C(N2CC(C)(NC(C3CC3Cl)=O)C2)=O)cc2cncc(Br)c2s1 CC1(CNC(c2scnc2C(F)(F)F)=O)CCN(C(=O)Cc2ncc(Cl)s2)C1 C1(NC(c2c(OC)nccn2)=O)CN(C(=O)CCCN2CCCCC2)CC1(C)C c1(CC)cccc(CC)c1C(N1CCN(C(C2(C#N)CCCO2)=O)CC1)=O C(=O)(C(C)S(C)(=O)=O)NCC(C)(Cn1cccn1)NC(C(C)CF)=O N1(C(C(C(C)(C)C)C#N)=O)CC2(CCCN(C(C3CS(=O)(=O)C3)=O)C2)C1 c1(C(=O)NCC#CCNC(=O)CSCC2CCCO2)cc(C2(C)COC2)no1 Cc1n[nH]cc1CNCC(C)N(C)C.C12(CCCC1)C(=O)NC2 C1(C(N2C(CC(=O)OC)CCC2)=O)CN(C(=O)CCCOC(C)=O)CCN1C c1(C(=O)NC2CCN(C(=O)C(C3CCOCC3)O)CC2F)cccn2nnnc12 Cc1ccc([N+](=O)[O-])c(C(N2CCC(NC(=O)Cc3conc3C)C(C)C2)=O)c1 CCC(C)(CNC(=O)NCCCCn1ccc(C)n1)C(N)=O c1(CC)[nH]nc(C(=O)NC2CC23CC(NC(c2ccc(COC)[nH]2)=O)C3)c1Cl c1(CCC(=O)NC(C(C)NC(COCCSC)=O)CO)c(F)cccc1Cl c1(N(CC)Cc2ccc(C(N)CN3CCCCC3)cc2)cnc(Br)c(Br)c1 CCCCC(CC)C(=O)NCC(CNC(=O)CNS(=O)(=O)N(C)C)CO Cc1ncc(C=CC(=O)NC2CN(C(=O)CC(C)(O)C3CC3)CC2C)s1 Cc1cc([N+](=O)[O-])ccc1N1CCC(C)C(N(C(C2CC2(C)C(C)C)=O)C2CC2)C1 C1(CCC)CN(C(c2ccnn2CCC)=O)CCN1C(C1CC=C(C)CC1)=O C1(NC(CN(CC)CC)=O)CN(C(=O)CC2CCCC2)CC1O C(CN=c1[nH]cnc(C)c1C#N)C1CC(NC(CC(CC)CN(C)C)=O)C1 C1(NC(C2(C#N)CC2)=O)CN(C(C2CCS(=O)(=O)C2)=O)CC1CC(F)(F)F CCN=c1ccc(C(N2CCCC2CCNC(c2cnn3ccsc23)=O)=O)c[nH]1 N1(C(CCc2nc(C)sc2)=O)CCC2CN(C(=O)CSC3CC3)CCC12 C1(CNC(c2n(C)ccn2)=O)CN(C(=O)C=C2CCOCC2)CCCO1 c1(C(=O)NCC2N(C(C(CC=CCC)C)=O)CCC2)ccc(OC)c(N)n1 C1(C)(CC(C)C)CCN(C(=O)C(Cn2cncn2)NC(=O)CNC(N)=O)C1 C(=O)(C1=NOC(C)C1C)N1CC2C(NC(CCOC)=O)C2C1 C1(NC(COCCOC)=O)CC12CCC(NC(=O)COc1ccc(Cl)cn1)CC2 CCC(CC(=O)NC(C)(C)CCCC(=O)NC(C1CCCCC1)C)CC(C)C C1(CNC(=O)C(O)C2CCC2)CCN(C(C2CCS(=O)(=O)C2)=O)C12CC2 CC1CCc2sc(C(=O)NC3(CF)CCN(C(C4COC(=O)O4)=O)C3)cc2C1 Cc1ccc(Cl)c2[nH]c(C(=O)NC(C)CCNC(=O)CNc3cccnc3)cc12 CN1C(=S)NC(c2nccc(Cl)c2Cl)C2=C1CN(c1ccc(F)cc1)C2=O C1(NC(C2CC(C#C)(O)C2)=O)CCN(C(C2(CC)CCNC2=O)=O)CC12CCC2 C1(C(=O)NCCCCO)CCC(n2cc(-c3cncc(Cl)c3)nn2)CC1 C1(CC)CN(C(=O)CCCC2CC2)CCN1C(C1CCC(F)(F)C1)=O C(=O)(CC1=CCCCC1)N1CCCC(CN(C)C(C2COCCOC2)=O)C1 N1(C(c2cc(C)ncc2)=O)CC(NC(c2csc(Br)c2)=O)CC(C)C1 C1(C)(C(N(C2CN(C(CNC(C(CC)C)=O)=O)CC2O)C)=O)C(C)(C)C1(C)C CN1CCOCC1CCC(=O)NC1CCCN(C(c2cncc(C(F)F)c2)=O)C1 c1(C(N(CCCCCNC(C2(SCC)CC2)=O)C)=O)c(S(N)(=O)=O)cnn1C c1(COC)nc(C)c(C(N2CC3CC2(CNC(C2CCCCS2)=O)C3)=O)s1 N1(C(C2N(C)CC(C)(C)C2)=O)CCC(C(N2CCCC(F)(F)CC2)=O)C12CCC2 C1(CC(N2C(C=C)C2)=O)COC2(CCC2)CN1 c1(C(C)OCC)nc(C(=O)N(CCNC(=O)C(F)=C(C)C)CC)cs1 C(C(C)(C)CC(=O)N1CC(F)CC1CNC(=O)C(c1cccc(C#N)c1)C)OC Cc1oc(Cl)nc1C(=O)NC(CNC(C12COC(CF)(C1)C2)=O)C1CCC1 c1(NC2(CNC(N3CCN(CCCC)CC3)=O)CCC2)cc2ccccc2[nH]1 N1(C(CCC=CC)=O)CCN(C(=O)C(C(C)C)c2ccn(C)n2)C(C)C1 c1(SC(C)C)nnc(CN(C(C2(SCC)CC2)=O)C(C)C2CC2)o1 C1(C(=O)NCC(C)C(=O)NCCN2CCC(CO)C2)(OC)CCC(C)C1 c1(C(N2CC(O)(CNC(C(C)CC3CCC3)=O)C2)=O)noc2c1CCCCC2 N1(C(c2n(C)c(Cl)cn2)=O)CC2CS(=O)(=O)CC2(NC(C23COCC(C2)C3)=O)C1 C1(NC(=O)COc2ccon2)CC2CCC1CN2C(=O)COc1n[nH]cc1Cl c1(C(N2C(CN(C(c3csc(C)c3N)=O)C)CC(F)C2)=O)nnc2n1CCCC2 C1(NC(c2cn(C)nc2O)=O)CC2(CCN(C(c3nonc3N)=O)CC2)C1 c12cccc(c1)NC2=O.C1(C(=O)NCCC)CCN(C(=O)C(C)SCC)C1 C1(C(N2CC(C)(NC(C(C)=C3CC3)=O)CC2(C)C)=O)C2C3CC4C1C1C2CC3C41 C1(NC(c2nn(CC)c(O)c2)=O)CCCN(C(c2cc(OC)ns2)=O)C1COC C1(c2nnnn2C(C)C)(NCC2C(OC)OCC2)CCC(CC2CCCO2)CC1 Cc1cnc2cc(C(=O)NC3CCC3NC(c3cc(C(F)F)ccn3)=O)ccn12 C(=O)(C1=CCCCCC1)NC1CCN(C(c2c(Cl)cn(CCC)n2)=O)CC1CC C1(C(=O)NC(C2CN(C(=O)Cc3cnnn3C)CCO2)C)CN(C)C(=O)N1 C1(C(N2C(CNC(C=CCC)=O)CC2)=O)CN2CCCN1CC2 C(=O)(C(=O)N=S(C)(C)=O)NCc1c(CC)cncc1.C123CC(C1C2)n1cc(nn1)C3 Cc1ccn(C)c1C(N1CC(NC(c2cc(C(=O)N(C)C)no2)=O)C1)=O CC1=C(C)CC(C)(C(=O)NCC23CCC(CC2)N3C(C2C3CC(=O)CC23)=O)CC1 C1(CCC)CN(C(=O)CN(CCCOC)C)CCN1C(=O)C(F)C1CCC1 c1(C(N2CC(CNC(CCC=C=C)=O)C3C2C3)=O)ccc(OC)c(F)c1F N1(C(c2cc(C)nn2C(F)F)=O)CCC2CCN(C(c3cnoc3)=O)CC2C1 C1(CNC(CC(C)NC(Cc2nc(C)oc2)=O)=O)CCCC(CO)C1 C1(CN(C(c2c(C(C)C)nns2)=O)C)COCCN1C(C1CCCCC1)=O c1(NC(C2(N)CC2c2nn[nH]n2)=O)ccc(I)cc1 C12(CNC3CN(C)CC3(C)C)CC3CC(C1)CC(N)(C3)C2 C#Cc1ccc(Cl)c(C(=O)NCC2CCN(C(C3COCCN3C)=O)C23CC3)c1 C1(NC(COc2cc(C)on2)=O)CCN(C(c2ccn(CCO)c2C)=O)C1C N1(C(C2CCCC(OC)C2)=O)CCCC(O)(CNC(C2CC3CCC2CC3)=O)C1 C1(C(=O)NCc2cccc(NC(C(n3ncc(C)c3)C)=O)c2)CCN(C)C(=O)C1 c1c[nH]cc1C(C)C.C12CC(C1)C(=O)NCCOCCN(C)C(=O)C2.C(C)(C)S CC(O)CCCN(C)C(C1(CCNC(=O)CC=CC(C)(C)C)CC1)=O C1(CCN(C(=O)OC(C)(C)C)CC(=O)CCCOC(F)F)C(Cl)(Cl)C12CC2 c1(N2CCCC(CCNC(C3CCC=CO3)=O)C2)cc(C(F)(F)F)nc(Cl)n1 C1(CC(=O)NC2CC(CNC(CN(S(C)(=O)=O)C)=O)C2)NC(=O)CN(C)C1=O CC1(C)CC(C(=O)NCC2(C)CC3CC3C2)CN1C(=O)Cn1cncn1 c1(NCC(CC)CC(F)(F)F)ccc(S(=O)(=O)NC2CCCCC2N(C)C)cn1 c1(C(N2CCN(CC(C)O)CC2)=O)nc2ccc(Br)cc2s1 c1(C(=O)OC)c[nH]c(=NCCNC(C2CCCN2Cc2ccccc2)=O)cc1C CC(C)CCCCCC(=O)N1CC(NC(=O)CS(N)(=O)=O)C(C2CC2)C1 C1(C(=O)O)CC2CN(c3nc(CO)ns3)CC2C1.CC(C)(C)C(=O)NC(C)(C)C c1(C(=O)NCCC(=C)CNC(c2ccc(C)nc2)=O)ccccc1SC(F)F c1(OC)cncc(N(C(c2nc(Br)cn2C)C(=O)NC(C)C)Cc2ccccc2)c1 C1(N(C)C(c2cnc(N)cn2)=O)CN(C(=O)Cc2ccccc2Cl)CC1(C)C c1(OC)cc(Cl)ccc1NC(=O)CCC(C)(C)C.N12CC3CC3(C1)C2=O C12(OC)CCC(CC1)N(C(C1CC3CN(C(C4CC=CC4)=O)CC3C1)=O)C2 c1(C(=O)NC2CCC(OC(c3conc3C)C)C2)cc(F)cc2c1NCCC2 c12cccc(n1)CN2.N1(C(C2C(C(=O)OC)C2)=O)CCN(CCF)CC1 N1(C(c2c(OC)ccs2)=O)CCC(CNC(c2ncc(N)cc2Cl)=O)C(F)(F)C1 N1(C(c2c(C)scc2)=O)CC(N(C(=O)C(C)CSCc2ccccc2)C)C(O)C1 N1(C(C2(COC)CC2)=O)CC2(CCCC2NC(=O)CC(C)P(C)(C)=O)C(C)C1 N1(C(C(CC[S+](C)C)O)=O)CCCC2(C1)CN(C(=O)COCC1CCOC1)C2 c1(C(=O)NC2CC(C)(NC(CSC)=O)C2)cnn(C)c(=O)c1 C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1(CC)CCCN(C(c2c(C#C)c[nH]n2)=O)C1 c1(OC)ccc(C(N2CCCCC2CCNC(C2(OC(C)C)CCOC2)=O)=O)nc1 CC(=O)CCCCC(=O)N1CCCCC(CNC(=O)CCCCCN(C)C)C1 N1(C(c2cc(Br)ccn2)=O)CCC(F)(C(=O)NCCCCn2ccnc2)C1 Cc1cnn(CCCNC(=O)CC2CC2)c1.C1(NC=O)CC(CF)C1 C([N+](=O)[O-])NCC(=O)NC1C(CNC(C2C(C(=O)OC)C2)=O)C1 n1(CC(=O)NC2CN(C(=O)CCC3CC3)CC3(CC3)C2)ncc2ncccc12 C1(C(=O)NCCCN(CCO)CCO)CC(F)(F)CN1C(c1csc(CO)n1)=O N1(C(C(=O)NCCC)C2CC2(Br)Br)CCN(CC(c2ccccc2)=O)CC1 C=CCC(CNC(=O)CCCSC1(C(C)(C)OC)CCCC1)NC(N)=O C1(CNC(C(COC)C)=O)CN(C(=O)CC(C)(F)F)CC2(CCC2)O1 c1(C(=O)NCC2CC(C)N(C(c3ccc(O)c(F)c3)=O)C2)cccc2[nH]ncc12 C1(NC(C2CCCO2)=O)CS(=O)(=O)C12CCN(C(=O)C=CC1CCCO1)CC2 C1(CNC(CCc2cnc(C)s2)=O)CC2(CC(NC(=O)C(C)c3ccco3)C2)C1 c1(C(C)=O)ccc(C(N2CCC(CNC(C3CCCN3C(C)C)=O)C2)=O)cc1C c1(C(=O)NCC2C(CNC(c3ccc(O)cn3)=O)C2)cc(Br)cc(F)c1F C#Cc1cc(C(=O)NC(CNC(=O)C=C(CC)CC)CC(F)(F)F)ccc1Cl Cc1sc2ccccc2c1C(=O)N(CC(O)CNC(c1cnco1)=O)C Cc1cccc(C(N2CCC(C(=O)N(CC(O)CO)CCO)C2)=O)c1F N1(C(CC2C(C)(C)CCO2)=O)CCCC2(NC(c3cncc(F)c3)=O)CC12 C=CC1(C(N2CCC(CNC(c3ccc(C)cc3N)=O)C2)=O)CCOCC1 C(=O)(C(F)(CNC(=O)C(C)(C)OCC)C(C)C)NCCOCC N1(CCNC(CNC(CNC(c2c(C)noc2)=O)=O)=O)CCCC(C)C1 c1(CNC(=O)NC(C(C)C)C2CCCO2)nc(-c2ncccn2)no1 c1(OC(c2nnc(-c3ccc(Cl)cc3)o2)C)cc(Cl)c(C(F)(F)F)cc1F C12(NC(CCCC(=O)NC)=O)CCCN(C(c3ccc(F)c(F)c3)=O)CC1C2 C(=O)(CC1=Cc2ccccc2C1)NCC1CC(OC)CN1C(C1CCC(O)C1)=O N1(C(C(=O)OCC)=O)CC(C(=O)Nc2cnc(C)c(OC)c2)OC2(CCC2)C1 N1(C(C(C)C(C)(F)F)=O)CCCC2(C1)CN(C(=O)CCCc1cnn[nH]1)CCO2 c1(N2CCCC(O)CC2)nc(=NC2CCC(F)(F)C2)[nH]c2c1CCC2 Cc1cc2cc(C(=O)NC(C)(C)C(C)NC(=O)C#CC3CCOC3)ccc2cn1 c1(CC(=O)NCCC2CCN(C(c3cc(C)c(C)o3)=O)CC2)cn2ccsc2n1 CC(C)C(C)(CNC(c1cnn(C)n1)=O)NC(=O)C=Cc1cn(C)cn1 C(=O)(CC(C(F)(F)F)c1ccccc1)NCC(=O)OCCC CC(C)(C(=O)NCc1nocc1C(=O)NCc1cscn1)n1cnnn1 c1(CC(=O)NC(CNC(C2(COC)C=CCC2)=O)(C)C2CCC2)cccnc1C N1(C(c2n(CC)cnn2)=O)CC2(CCN(C(=O)CC3CCCNC3=O)C2)C1 C(=O)(CCS(=O)(=O)N(C)C)NC1CN(C(CCCCC)=O)CC1CO C(CC(C)C(=O)NCC1CN(C(c2cc(C(=O)OCC)c[nH]2)=O)C2CC12)=CCC Cn1ncc(C(N2CCC(CCNC(=O)CCc3c[nH]c(=N)[nH]3)C2)=O)n1 Cc1ncsc1C=CC(=O)Nc1cccc(CNC(C2CCCS2)=O)c1 C(CCN(C(=O)Cc1csc(Cl)c1)C)(C(C)(C)C)NC(C1(COC)CCOC1)=O C1(CN(C(C(CCSC)NC(N)=O)=O)C)CCCCN(C(=O)CSC(F)F)C1 C1(C(N2CC(NC(c3ccn(C)n3)=O)C(CO)CC2)=O)COc2ccccc2C1 C(c1ccccc1)=C(C(=O)NCC1(N(C(=O)COC2CC=CC2)C)CC1)OC N1(C(C(c2ccc(Cl)cc2)C)=O)CCC2(CCCN2c2ccnc3ncnn23)C1 N1(C(C=CC(N)=O)=O)C2CCC1C(NC(=O)CCCn1cncn1)C2 c1(C(N2CC(NC(C(CC)SC)=O)C2)=O)cnn(-c2ccccc2C)c1N.C(C)C N1(C(CCN(C)CC)=O)CC2CCC(N(C)C(c3cc(C)cc(Cl)c3)=O)C2C1 c1(CC2C3CN(NCC4CCC(CCCC)O4)C2CC3)cc(F)cc(C)c1N c1(C(=O)NC(CNC(C(CC)NC(C)=O)=O)C)cccc(OC2CCCCC2)n1 c1(N)ncccc1C(F)(F)F.n1(CC(=O)NC2(COCC)CC2)nnc(C)n1 C(=O)(C1=NOC(CNC(=O)C(=O)NC2CC2)C1)NC(COC)C1CC1 C1(CC(=O)NCC(C)NC(C(C2CCOCC2)C)=O)CC2CCC1O2 Cc1ncc(NC(C2CCCN(Cc3cc(-c4ccco4)on3)C2)=O)nc1C c1(C(N2CCC(N(S(C)(=O)=O)CC)C2)C(=O)NC2CCOC2)sc(Br)nc1C c1(N(c2cc(OC)c(C)cc2)CC2CNCCCO2)ncnc2cc[nH]c12 c1(NC(c2n(CC=C)nnn2)c2cncn2C(C)C)cccc(OCC(F)(F)F)c1 C1(CNC(CCCOCC)=O)CCN(C(c2c(C)noc2C(F)F)=O)CC1(F)F CN1CCC(CCC(=O)NCCSCC(=O)Nc2cccnc2)CC1 C1(CNC(CC(C)(F)F)=O)C(C2CC2)CCN1C(=O)Cc1nc(C2CC2)nn1C n1(CC)nc(-c2ccccc2)cc1C(c1ccccc1)NCC(C(=O)OC)OC CC1(C(N2CCC(CCCO)CC2)=O)CCCN(C(c2cnnc(O)c2)=O)C1 C=C=CCCC(=O)N(CCCNC(C1(c2ccccc2)CC1)=O)CC1CCCC1 C1(C(N(C(C)CNC(=O)C=CCOCC(F)(F)F)CC)=O)CCN(C)CC1 c1(N(CCC)C)ccc(C(N2CCCCC2CN(C(=O)C2=CCSC2)C)=O)cc1 N1(C(=O)C(C2CC(F)(F)C2)O)CCN(Cc2n(C)ccn2)CC1 CCC(CC)C(C(=O)NCCN(CCO)CCNC(c1cncc(C)n1)=O)OC N1(C(C=C(C)C)=O)CCN(C(=O)CC=Cc2ccc(F)cc2)CC1C CC12CC(C(=O)NCCCNC(C3CC(N(C)C)C3)=O)(C1)C1(CCC1)O2 FC(F)C(F)(F)CCN=c1ccnc(NCc2noc3c2CCCC3)[nH]1 C1(C(=O)Nc2scc(C(=O)OCC)n2)CCN(C(C)C(F)(F)F)CC1 C(=O)(C#CC1(C)COC1)N1C(NC(N2C3CCC(C(=O)OC)(C3)C2)=O)CCCC1 Cc1cc(C(N)=O)cc(CCNC(c2cc(Cl)c(Br)[nH]2)=O)c1 C#CC1(CNC(=O)C=CCC(C)(C)NC(C2CNC(=O)C2)=O)CCCC1 C12CC(=NO1)C(=O)N1CC(C(F)C1)NC2=O.C=C1C2C1C(=O)C2=O.OC.OCC N1(C(=O)CC2CCC(F)(F)C2)CC2CCN(C(C3CC=CC3)=O)CC(C2)C1 O=c1n(Cc2ccccc2)nc2ccccn12 c1(C(=O)NC(C(C)OC(CC(c2ccc(C)cc2)C)=O)=O)cc2sccc2cn1 N1(C(c2ccc(N(C)C)cn2)=O)CC2CS(=O)(=O)CC2(NC(c2cscn2)=O)C1 c1(C(N2CCC(C3N(C(C(C)C)=O)CC(C)C3)CC2)=O)ccc2c(c1)CNC2=O C1(CNC(Cc2ccc(C)nc2)=O)CCC(C)N(C(=O)C(n2nccc2C)C)C1 C12(C(N3CCC(C(C)(C)NC(CC(CC)OC)=O)C3)=O)CCC(C#N)(CC1)CC2 C#Cc1ccnc(C(=O)NCC(C)CNC(=O)Cc2cccc(C(C)C)c2)c1 CCC(CC(C)O)NC(=O)CCC1(NC(c2csc(O)n2)=O)CCCC1 C(=O)(C1=C(F)CN(C(=O)CCCC(C)=O)CC1)NC(CCC)CC C1(C(C)C)CC(CC(=O)NCC2CCN2C(c2cscn2)=O)CCO1 c1(C(N2C(C(=O)NC(C3CCNC3=O)C)CCC2)=O)cccc(O)c1 N#Cc1c(Cl)nsc1NCC1CCCCC1NC(C1CC12CCCC2)=O C1(C)(C(N2CC(CC)(NC(=O)Cn3ncnn3)C2)=O)Cc2ccccc2NC1=O C=CC(C)(O)CC(=O)N1CCC(N(C)C(c2ccc(C)c(CO)c2)=O)CC1 c1(C(=O)NC2C(C)N(C(C3CC4CCC3CC4)=O)CC2)cncc(F)c1Cl Cc1ccc(N)cc1C(N1CCC(NC(=O)CCF)C(O)C1)=O N1(C(C2CC(C)N2C(c2cc(Cl)cs2)=O)=O)CCc2cnccc2C1 N1(C(C2N(C)CCC2)=O)CCC2CN(C(C3CC(C)(O)C3)=O)C2C1 c1(C(=O)NC(C(C)NC(C(CC#C)O)=O)(C)OC)ccc(OC)nc1F N1(C(C(C=C=C)C)=O)CCN(C(C2(CC)CC(=O)C2)=O)CC1C C1(C(=O)NCC(Cc2ccccc2)OC)C=CC(NC(c2ccncc2)=O)C1 N1(C(Cc2n(C)ccc2)=O)CCN(C(=O)C(F)=C2CCCC2)C2CCCCC12 c1(OC)ccc([N+](=O)[O-])cc1NC(C1COCCN1Cc1cnc(Cl)c(Cl)c1)=O C1(NC2(c3n(C(C)C)nnn3)CC3COC2C3)CC2C(=O)NCC(=O)N2C1 Cc1cc(C(=O)NC(C)CCCNC(=O)CNc2ccncc2)c2c(c1)CCC2 C(=O)(C(CCC(C)(C)C)N1CCOCC1C)NCCCSC c1(-c2ccc(OC)nc2)cccc2[nH]c(C(=O)Nc3c[nH]nc3Br)cc12 C(=O)(C(CNC(c1cc(F)ccc1C)=O)C(C)(C)C)N(CC(CC)C)C C(CN=c1ccc2nnc(-c3cccs3)n2[nH]1)NC(=O)CN1CCCCC1 C1(C(N(C)CC2CN(C(=O)COCCCN(C)C)CCO2)=O)CC2(C1)CC2(F)F n1(CC)cc(C(N2CC(C(N)=O)(CNC(C3CC4CCC3C4)=O)C2)=O)c(C)n1 N1(C(c2cc(C)sc2C)=O)CC(=O)NC2CN(C(=O)C(C)c3cc[nH]n3)CCC12 c1(C(N2CCC(N(C(=O)C(C3CC3)SC)CC)C2)=O)cc2nc(C)cc(C)n2n1 Cc1noc(C)c1CC(=O)NC(C)C.n1(C2(C)CC2)cc(CC(O)C2CC2)nn1 C1(C(N(CCOC)CCNC(=O)C(c2ccc(C)cc2)C)=O)COC2(CCC2)C1 CC(O)C(C(=O)NCCCNC(=O)CC1(C)CC(F)(F)C1)NC(=O)OC(C)(C)C N1(C(CC(C)(C)C)=O)CC(NC(=O)CC2CC(=O)NC2=O)CC2(CCOCC2)C1 N1(C(C(C)n2ccnc2)=O)Cc2n[nH]cc2C1C(=O)NC1C(C)C1C N1(C(C2C(CNC(C3CC(N4CCCC4)C3)=O)C2)=O)CCCC1CO N1(C(Cc2c(C)nc(C)s2)=O)CCC(NC(c2ccoc2Br)=O)C(F)C1 C1(NC(Cc2cc(C)[nH]n2)=O)CC2(CCN(C(c3ccc4c(c3)COC4)=O)CC2)C1 Cc1nc2cc(Cl)c(NC(C34CC3CN(Cc3cnc(O)nc3O)C4)=O)cc2o1 CC1(C)CC2(NS(C)(=O)=NC(=O)c3cccc(Br)c3)CC1C2(C)C C12(C(=O)NCCN(C(CC3CC(=C)C3)=O)CCC)CCCCC1OCC2 N1(C(c2c(CC)nco2)=O)CC(O)CC1(C)C(=O)NCc1cccc(O)c1C C1(C(=O)NC2CN(C(C(CC#C)(C)C)=O)CC2(C)C)CCn2cc(C)nc2C1 c1(C(=O)NC(C(=O)OC)Cc2ccccc2)cc(C(C)C)n(-c2ccccc2)n1 N1(CC(=O)NC2C3N(C(C(C(CC)C)C)=O)C(CC3)C2)CCCCCCC1=O N1(C(C)(C)C)CCCC(N2CC3CC(NC(C4CCCCC4(F)F)=O)C3C2)C1=O C12(C(C3CCCCC3)NC(Cc3scc(C)c3)=O)CCC(C1)C2(C)C C(=O)(CS(=O)(=O)CCOC)NCCC(=C)CNC(c1ccc[n+]([O-])c1)=O N1(C(CN(C)C)=O)CCC(NC(c2ccccc2OC2CC2)=O)C(CO)C1 c1(CC(=O)NC2C3CN(C(CCCCCOC)=O)C(C3)C2)cccc2nsnc12 C1(CNC(CC2(OC)CCC2)=O)CCC(C)N(C(=O)CCCC2CCCC2)C1 C1(CC(N2C(C)(C)CCC2)=O)CC2(CC2)CN1C(c1ccc(F)cn1)=O N1(CCC)C(=O)CCC1C(=O)NC(C)CC(C)NC(=O)C(C)C1CC1 N1(C(CCCOCC)=O)CC(NC(c2cc(C(C)(C)C)oc2C)=O)C2CC12 c1(C(=O)NCCC2CCN(C(CC=C)=O)C2)c[nH]c2ccc(F)cc2c1=O c1(OCC(N2CCC(NC(c3nnc(C)o3)=O)C2)=O)cccc(F)n1 C1(C(=O)NCCCOCCNC(CCCn2ccc(C)n2)=O)CCC2C1C2(F)F c1(C(=O)NC2C(CNC(c3ccn(CCOC)n3)=O)CCC2)cccc(F)c1F c1(N(CC)CC2CCSC(c3cccnc3)C2)ccc([N+](=O)[O-])c(OC(C)C)c1 C(C(C(C)C)C(C)C)NC(CCN(C(=O)Cc1ccccn1)CC=C)=O N1(C(C(C=C)(C)O)=O)C(CNC(C2C3CCCC23)=O)CC2COCC12 N1(c2c(C)cncn2)CC2CC1CN2C(c1ccn(-c2cccc(F)c2)n1)=O c1(NC(CN(C2CC(C#N)C2)C(COCC(=O)OC)=O)=O)csc(S)n1 N1(c2nnc(-c3c(OC)ccs3)o2)CCCC2CC12 C(=O)(CCCC(F)F)OCCO.CCCCNC(=O)CSC(F)(F)F C1(CC(=O)N(C(C)CNC(=O)Cc2sccc2C)CC)CC(C)=NO1 C1(NC(=O)OC)CCN(C(c2cn(CC3CC4CC4C3)nn2)=O)C1C(C)(C)C C1(OCCOC)CCN(C(C2CCCN2C(C2CC=CCO2)=O)=O)CC1 CC(Cn1ccnc1)N=c1[nH]c(=NCC2CCC=CO2)c2[nH]ccc2[nH]1 C1(CNC(C2C(C)CC3CC3C2)=O)CCN(C(=O)C(F)C(F)(F)F)C1(C)C C1(N(C(C2(C#N)CCC2)C(=O)NC)C)CCCC(C(=O)OCC(C)(C)C)C1 N1(C(CCNC(C)=O)=O)CCC2(NC(=O)Cc3nnc(C)o3)CCCCCC12 C1(C)(CNC(CCOCC)=O)CCN(C(=O)CC2(OC)CCCCC2)C1 C12C3CC4CC1CC(C4)(C3)CC(=O)NC2.CC1(C)C(CO)CC1O c1(OC)ccc(CNC(=O)C(c2nncn2C)N(C(C)C(C)C)C)cc1 Cn1cncc1-c1cn(C2CCN(C(=O)C(C)(O)c3ccccc3)C2)nn1 c1(OC)cnccc1C(N1CCC(C)C1CNC(=O)CCc1ccc(C)s1)=O Cc1ccc(C(C)CC(=O)NCCCCn2cc(C(C)N(C)C)nn2)cc1 C1(C(=O)NC(CC=C)CNC(c2ccc[n+]([O-])c2)=O)CCn2ncnc2C1 N(C(=NCCF)N1CCC(c2csc(C)c2)C1)C(CC)Cc1ccc(Br)cc1 N1(C(=O)Cc2cc(Br)cs2)CCCC(C2CN(C(C3OCCO3)=O)C2)C1 C1(C(=O)NC2CCCC2NC(C2CCOC(=O)N2)=O)(OCC)CCOCC1 C1(NC(=O)C=CI)CCC2CCN(C(c3cc(O)nc(O)c3)=O)C1C2 CC1(CCO)CCN(C(C2(NC(=O)CN3CCC(F)CC3)CCCCC2)=O)C1 CCC(C)C(O)C(=O)NCCCCCCN(C)C(c1ccn(C)n1)=O C(C)(CC(N)=O)NC(CCNC(C(C)NC(C)=O)=O)=O c1(C(N(CC(C)NC(c2scnc2C(C)(C)C)=O)C)=O)ccc(F)cn1 Cc1c(C(N2CCC(C(N3CCOC(C#N)C3)=O)C2)=O)cccc1F c1(C(=O)NC2CN(C(c3c[nH]c(=NC)o3)=O)CC2(C)C)ccn2c1CCCC2 C=C(C)CC(C(=O)N(CCOC)CC)NC(c1n[nH]c(C)c1O)=O c1(CC(=O)NC2CC(C(F)Cn3cc(-c4ccccc4)nn3)C2)cccnc1Cl C12CCN(C1)C2=O.n1(CC(=O)NC2CCC2C(F)(F)F)cnnn1 N1(C(C)=O)CCC(CCC(C)(C)NC(=O)CCc2ccsc2)CC1 C1(C(=O)NC2CCC2)CN(C(=O)C=Cc2cocn2)C2(CCC2)C1 c1(N2CCC(CN(C)CC)CC2)cc(NC(c2ccncc2F)C)nc(C)n1 C1(C(C)NC(=O)CCC2CC2(C)C)CCN(C(c2c[nH]cc2Br)=O)C1 C12CCCC1CNC(=O)C(C)OC2.c1(CC(=O)NC2CC2)ccccc1 CCS(=O)CC(=O)NC(CCN(C(=O)C=Cc1cn[nH]c1)C)C(C)C C#Cc1ccc(F)c(NC(C)CCN(C)C(=O)OC(C)(C)C)c1 c1(CNC(CC2C(CNC(c3c(CC)ncnc3)=O)C2)=O)ccc(F)c(O)c1 N1(C(C(CC)=CC)=O)CC(CNC(=O)Cn2cc(C3CC3)nn2)C(C)(C)C1 c1(C(=O)NC(CC)CNC(c2cc(C)on2)=O)ccc(S(N)(=O)=O)s1 Nc1cc(C(=O)NC2CCN(C(=O)C(CO)c3ccccc3)C2)ccc1Cl c1(CC)ccc(CC(N2CCCC(NC(c3csc(CC(C)C)n3)=O)C2)=O)cc1 Cc1cc(OCC(N2CCN(C(c3n[nH]c(O)n3)=O)CC2CCO)=O)cc(C)c1 N1(C(N(OCCC(C)C)C(C)C)=O)CCC2(CCCNC2=O)CC1 N1(N(C)CP(C)(C)=O)CCCC12CCCOC2.C(=O)(CCS(C)(=O)=O)C1NCC1 c1(NCC(=O)NC23CC(C(=O)NC4CC4)(C2)C3)ccc([N+](=O)[O-])cn1 c1(C(N2CC(COC)N(C(=O)Cc3cncs3)CC2)=O)cc(Cl)cc(C)c1N C1(CNC(CC=C=C)=O)CC(C(F)(F)F)CCN1C(=O)C(CC1CC1)CC1CC1 C(=O)(CN=c1cc[nH]cc1)N1CC2C(NC(C3CC34CCC4)=O)C(C2)C1 C1(C(=O)NCCNC(CC2(C)CC2)=O)CN(C(c2cc[nH]n2)=O)C1 c1(NC(CCN(C(C(CN(C)CCO)O)=O)CCO)=O)ccccc1N C1(NC(Cc2ccc(C)s2)=O)CC2CN(C(=O)CC(C)C)CCN2C1=O CC1=C(C(=O)N2CCC(C)(C(=O)NC3CC3C(C)C)CC2)CCO1 N1(C(c2cc(=N)[nH]cc2)=O)CCCC2C1CCCN2C(=O)Cn1c(O)nnc1O N1(C(C2C(C)N(C(c3cn(C)cn3)=O)CC2)=O)CC2(CCC1CO)CC2 Cc1cn(C)nc1C(=O)NCC1(CNC(c2ncccn2)=O)CCC1 N1(C(c2cc(C)n(C(C)C)n2)=O)CCC2OCCN(C(C3CCC(C)O3)=O)C2C1 N1(C(COc2c(C)ccc(Cl)c2)=O)CCc2sc(S(N)(=O)=O)cc2C1 C(=O)(C1CCCc2cccnc21)NCC(C)NC(=O)C1=CCCCCC1 C1(N(C)C)CC2(CCC(C(N3CCCC(NC(C4CCCCO4)=O)C3)=O)CC2)C1 C1(CC(=O)NC2CCN(C(C(C)(C)CC#N)=O)C2)Oc2ccccc2NC1=O Cc1nc[nH]c1CC(=O)NC1CC(C)(NC(=O)C(C)OCCC(C)C)C1 c1(C(N2C3CN(C(CCC(=O)OCC)=O)C(C3)C2)=O)ccc2c(c1)N(C)C(=O)C2 C(C(O)CN=c1cc[nH]cc1C#N)NC(C(C)SC)=O CC1CCCCN(C(c2cn(CC(F)(F)F)cn2)C(=O)NC2COC2)C1 Cc1cn2cc(CC(N3CCOC(c4ccc(F)cc4F)C3)=O)nc2s1 C=CCCC(CC(C)C)C(=O)NCC1(NC(c2ccnc(F)c2N)=O)CC1 C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)(CC2CC2)CCCC1 Cc1ccn(CC(=O)NC(CNc2cccn(C)c2=O)C(C)(C)C)c(=O)c1 c1(C(=O)NC2CCN(C(C3C(C=C)C3)=O)C2CC)sc2cc(Cl)ccc2c1Cl C12(NC(C)=O)CC(N(c3ccccc3)C(C3(CNC)CC3)=O)(C1)OC2C.C(C)(C)N C(=O)(CC(C)(C)CC(F)(F)F)NCCN(C(CCC(c1c(C)n(C)nc1)=O)=O)C Cc1nc2n(n1)CCN(c1ccnc(N3CC4(COC4)C3)n1)C2 n1(CCC(N2CC(COCC)OCC2)=O)c(C)nc2ccccc12 CCCCCC(C)CC(=O)NCC1CCCC2(CN(C(=O)C(O)COC)C2)O1 CCCC(C)(O)CC(=O)N1CC(NC(c2coc(CC)n2)=O)CC(F)C1 C1(C(=O)NC2C(NC(c3c(C)con3)=O)C2)CCc2c[nH]nc2C1 N1(C(C(CC)C)=O)CCC(CCN(C)C(c2coc(Cl)n2)=O)CC1 C1(N(C)C(c2cnc[nH]2)=O)CC2CCC(C1)N2C(c1cnnc(O)c1)=O N1(CCNC(c2c(CCNC(C(C)NC=O)=O)ocn2)=O)CCC(O)CC1 N1(C(C2C(C(=C)C)OCC2)=O)CCC(C(N2Cc3cncnc3C2)=O)CC1(C)C N1(C(c2cc(C(N)=O)no2)=O)CCC2CN(C(=O)C=Cc3ccncc3)CC12 c1(OC)cncc(C(N2CC(NC(=O)CC(C)(C)C3CC3)C2)=O)c1 C1(NC(C(CC)F)=O)CN(C(C2(C#N)CC(=O)C2)=O)CC2(CC2)C1 CCCCC(O)C(=O)N1CCCC1(C)CNC(c1coc(C(N)=O)c1)=O C1(C(C(=O)NC(CC)C)N(C)Cc2cccnc2)CCC2(CC2)C1 c1(OCC)cc(C(N2CC(OCC)C2)=O)oc(=O)c1.C1(=O)CC(C)N1.C1(N)CCCC1 c1(CC(C(=O)NCCN(C(=O)Cc2ccn(C)n2)C)OC)ccc(F)cc1 C1(CNC(C2CCN(C(C3(CC4CC4)CCC3)=O)C2)=O)CC1C1CC1 C(C(=O)N1OC2CCC1C2)N(C(CNC1CC(=O)C1(C)C)=O)CC#C C1(CC(=O)NC(CN(C(c2ncn(CC)n2)=O)CC)C)CCCC(=O)N1 Cc1cc(C(F)(F)F)cnc1Cl.C12CN(C(=O)CCCCCF)CCC1C(=O)N2 N1(CC(=O)NC2(c3ccncc3)CC2)CCN(C(=O)CCCC2CCC2)CC1 c1(NC(CC2C(C)(C)C(CNC(=O)CC3CSC3)C2)=O)cccc2c1CCC2 N1(C(CC(C(C)C)(F)F)=O)CC2CCC(C1)N(C(=O)C=CC1CCOCC1)C2 N1(C(CCC2CCCN(C(c3c(CC)c[nH]c3)=O)C2)=O)CC2CCCCC12C N1(Cc2cn(C3(N(C)C)CC3)nn2)CCCC(NC(=O)CC(C)N(C)C)C1 C=C(Cl)CC(C(=O)N1CCCC1Cn1ccnn1)NC(c1scnc1Cl)=O C1(NC(c2c(C)cccn2)=O)CCN(C(=O)CN2CCCCCC2=O)CC1F CC(=Cn1ccnn1)C(=O)NCCCCNC(C1SCCS1)=O C1(CC)(NC(=O)C(C)OCOC)CCN(C(=O)C=CCF)CC1 C1(C(N2CCC(CCNC(C34CCCN3CCC4)=O)C2)=O)C(F)(F)C12CCC2 C=CC(F)(F)C(=O)NC1CC(NC(c2csc(O)n2)=O)C1 c1(C(N2CCC(OCC)CC2C)C(=O)NC2CCOC2)cc2n(n1)CCCC2 C1(NC(C(C)=C(C)C)=O)CC2(CCN(C(C3(C(F)(F)F)CC(F)(F)C3)=O)C2)C1 c1(CNC(c2cccnc2)=O)ccnc(C(=O)NC(CC2CCCC2)CO)c1 c12ccc(cc1)NC1CCC(CC1)C(=O)NC(=O)CS2.c1(CC)ccc(C)cc1 CCC(CC)C(C(=O)NC1CCC(CNC(=O)C=CC=C(Cl)Cl)C1)OC C#Cc1cccc(C(=O)NC2CC(F)(CNC(=O)C(F)=CC3CC3)C2)c1 N#Cc1cc(C(=O)NC(C(=O)NCc2nc(C3CC3)no2)C2(O)CCC2)c[nH]1 C1(C2CN(C(C(C3(O)CCCCC3)NC(c3nc(C)sc3)=O)=O)C2)CC2C=CC1C2 CP(C)(=O)c1csc(C(=O)OCCOc2ccc(F)cc2Cl)c1 CCC(C)CCCCC(=O)NCCOCCN(C)C(c1cc(N)c(F)cc1F)=O C1(C)(NC(C2N(C(c3cc(C)n(C)c3C)=O)C(C)C2)=O)CN2CCC1CC2 C12CC(C1(C)C)OC(=O)CC2.n1(CCCC)cc(CNC(=O)NCC)nn1 Cc1ccc(N)c(C(=O)N(C(C)CCNC(=O)Cc2ccc(Cl)nc2)C)c1 c1(C(CN(C(=O)CN(CC(C)(C)C)C)C)NC(COC(C)=O)=O)ccccc1 CCCC(C(C)C)c1nc(C2CCOC2)nn1-c1ccncc1C Cc1ccc(CC(=O)NC2CN(C(=O)C(N3CCSCC3)C)CC2(C)C)c(F)c1 S(=O)(=O)(c1c[nH]c2ccc(Br)cc12)NC(c1ccc(N2CCOCC2=O)cc1)=O c1(C(=O)NCC2C(NC(C(C(C)C)SC)=O)COC2)c(O)ncc2c1CCC2 C1(CNC(CC2C(SCC)C2)=O)CCC(NC(=O)C(C)(C)n2cnnn2)CC1 CC(c1ccco1)=CC(=O)NCCCC1CCCN1c1ccnc(C2CC2)n1 c1(OC)cc(F)c(C(=O)NC2CN(C(=O)C=Cc3cscn3)CC2C)cc1N c1(C(=O)NCCC(O)C(=O)NCCc2ccccc2)ccc2cc[nH]c2c1 N1(C(C2CC3CCC2CC3)=O)CC2CC(NC(C3(n4nccn4)CC3)=O)CC2C1 C1(C(N2CC(O)(CCNC(C(C(C)C)NC(C)=O)=O)C2)=O)CCCC2C1C2(F)F C1(CC(=O)NC2(CNC(c3ccc(F)o3)=O)CCC2)CCCC12CC2 CCC(C)C(C)CNC(c1cc(CNC(C2CS(=O)(=O)C2)=O)nn1C)=O C1(NC(c2c(CCC)nns2)=O)CCC(C)(CNC(c2ccc[nH]2)=O)C1 Cc1cc(C)nc(N2CCN(C(c3cccc(O)c3F)=O)CC2CO)n1 c1(C(N2CCCC(NC(C3(CC=C)COC3)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(C)NCc2c(NC)nccc2)ccc(F)c(Br)c1 C12(OC)CCC(C(=O)NCC(C)NC(C3CC=C(C)CC3)=O)(CC1)C(=O)C2 N1(C(c2sccc2Cl)=O)CC2CC(C1)N(C(c1nc(C3CC3)ncc1Cl)=O)C2 Cc1nn(C)c(C)c1CCC(=O)NCC(O)CN(C)C(c1ncn(C)n1)=O N1(C(CCCC=C)=O)CC2CCCCC2(NC(=O)C(C)CCOC)C1 C=CCC(C(=O)NCCC1(O)CN(C(=O)C(O)CC(F)(F)F)C1)C(C)C n1(C(CC)C)nnnc1C(CCC1CC1)NCc1cocn1 C1(NC(C2(F)CCCOC2)=O)C2CN(C(c3ccn(CCF)n3)=O)CC12 c1(NC(N(C(c2ccc(OC)cc2)CO)C)=O)cc(S(C)(=O)=O)cc(Br)c1C c1(C(=O)NCC(C)NC(c2snc(C)c2N)=O)cc2cc(F)ccc2o1 c1(C(N2CC(CC=C)(C(=O)NC(CC3CC3)CO)C2)=O)cc2ccccc2[nH]1 N1(C(C2(CC#C)CCN(C(=O)C(F)n3ccnc3)C2)=O)C2CCCC1COC2 c1(SC)nc(=NC2CCCN(C(C34CCN(CC3)C4)=O)C2)c(C#N)c[nH]1 Cn1nc(Cl)c(C(=O)NCCCNC(=O)C(C2CCCCCC2)O)c1Cl c1(OC)c(Cl)ccc(Cl)c1C(=O)NC1CCC(F)(CNC(=O)CN2CC=CC2)C1 CN1Cc2ccccc2C(NC2CCCC2CN)C1 CCC(CC(=O)Nc1ccc[n+]([O-])c1)NC(=O)Cc1ccc(C)s1 C=C(C)CC(C(=O)NC1CN(C(c2ccc(Cl)o2)=O)CC1CCC)OC CCCCCCC(CC)C(=O)NCC1CCN(C(c2cnc3ccccn23)=O)C1 C1(C(=O)NCC2(OC)CC2)(NC(c2cscn2)=O)CCC1 N1(C(C2(F)C(C)C2)=O)CCC(n2cc(CNC(=O)Cn3nccn3)nn2)C1 Cc1ccc(C(=O)NC23CC(C(=O)NN4CCCCCC4CCO)(C2)C3)c(C)c1 C1(CC(=O)NC2C(C(=O)NCCOCCCC)C2(C)C)OCCC1(C)C C(=O)(C(CCC(C)C)NS(=O)(=O)c1ccccc1)NCCC(=O)OC C(C(F)(C(=O)NC1COCCC1CO)C(C)C)NC(c1c(C)con1)=O Cn1cc(C2CNC(=O)CCN(C)CCO2)cn1.CCC(=O)NCC1CC1.CO.CC C1(C)(CNC(C2(OC)CC(C)C2)=O)CN(C(C)=O)CC1C.C12CSCN1C2=O C(C)(C(C(=O)NCC1OCCC1(C)C)C(C)C)NC(c1c(NC)nccc1)=O C(C)(C)(CN=c1[nH]cnc(C(F)(F)F)c1C)NC(c1c(C)cccc1)=O c1(C(N2C(COC)CN(C(C3CCC3)=O)CC2)=O)ccc(Br)c(F)c1N c12ncoc1CNC2=O.C(=O)(C=CCNC(=O)OC(C)(C)C)NC(C)C Cc1ccc(CN2CCC(NC(c3oc(C(C)C)nc3C)=O)C(F)C2)c(O)c1 c1(OC)cnc(C(N2CC(NC(c3cccnc3)=O)C(C)C2)=O)c(F)c1 C#CC1(O)CC(C(=O)NCC(C)(C(C)C)NC(=O)C(=O)NC2CC2)C1 C(=O)(C(F)C(C)CNC(C1CC(F)CN1C)=O)NC(C(C(=O)OC)C)C CC1CCCCN1CCC1(CC(=O)NC(c2ccsc2Cl)=O)CC1 c1(NC(=O)Nc2c(C(=O)OC)cccc2)nccc(C#N)c1Cl C=C(C)CC(C)C(=O)NC(C)C(C)NC(c1ccc(OCC(F)(F)F)cc1)=O CCCCC(O)C(=O)N1CCC(C)(C)C1CNC(=O)CCc1ccc(CC)cc1 c1(C(=O)NCC(C)N(C(c2ccc(C(N)=O)s2)=O)CC)ccc(C2CC2)cc1 Cc1c(CC(N2CC(CNC(C3CC(=C4CCC4)C3)=O)CC2C)=O)cnn1C C1(NC(CC2(OC)CCCC2)=O)CN(C(=O)C(C)N=[N+]=[N-])CC1O C1(NC(CCC(=C)Cl)=O)CC2CC(C1)N(C(c1cccc(N)c1F)=O)C2 Cc1cn(C)cc1C(=O)NCCSCCCNC(c1ccc(C(N)=O)o1)=O C(Cc1cc[nH]n1)(C(=O)NCC1(O)CCOC1)NC(CC1C(C)CC1)=O C1(NC(c2nc(C#C)sc2)=O)CCCN(C(C2CC2(F)F)=O)CC1 c1(C(=O)NC(C)CNC(C23CC(C(O)C4CC4)(C2)C3)=O)ccc2c(c1)CCC=C2 c1(C(=O)NCC(C)CNC(=O)Cc2cnccn2)ccc(C(F)F)c(Cl)c1 c1(C(=O)NCCCNC(c2c(COC)scc2)=O)ccc(F)c(F)c1F N1(C(c2c(Cl)cn(C)n2)=O)CCC2(CC1)CN(C(=O)C1=CCC1)CC2CO c1(C(N2C(CNC(CCOC(C)=O)=O)CCC2)=O)cc(C(C)C)nn1C c1(C(C)(C)C)ccc(C(=O)NC(CNC(=O)CC2(C)CCOC2)CO)cn1 C1(CCOC)CN(C(=O)Cc2sccc2C)CCN1C(=O)C(=Cc1c[nH]cn1)F Cc1cc(OCCC(=O)NC(c2n[nH]c(C)n2)C)cc(C)c1 O=C(CC(C(F)(F)F)NC(c1ccc2[nH]ccc2n1)=O)NC1CCC1O C(=O)(C(C(C)C)N1CCN(C)CC1)N(CCNC(C(C)O)=O)CC1CC1 C1(C(=O)NC(CC)CN(C)C(C2CC2C2CCCCO2)=O)CCC(N(C)C)CC1 C(CNC(=O)CN1CCSCC1)(C(C)(C)C)NC(C(CC)Oc1ccccc1)=O c1(NC)cc(Cl)ccc1C(=O)NCCC(C(C)C)NC(c1cc[nH]n1)=O C1(NC(=O)CC2CCC(O)C2)CC2CC1CN(C(=O)CC1CC3CC3C1)C2 C(=O)(CC(C)CN(C)C)NC1(C)CC(NC(CC2CC(OCC)C2)=O)C1 c1(CCN=C(NCC2(C#N)CCC2)NC2CC2)ccc2c(c1)OCCO2 C1(C(N(CC(CN(C)C)O)C)=O)CCC(NC(C2CCCO2)=O)C1 C(=O)(C(C)C(O)C(C)C)N(C(C(C)C)C(=O)OCC1(NC(C)(C)C)CCC1)C1CC1 Cc1ccc(C(=O)NCc2c[nH]nc2C(=O)N(C)C)[nH]1.C12(CC1)C(=O)NC2 C1(CNC(C2C(CNC(=O)CCc3ccncc3)CCC2)=O)CCC(F)C1 N1(C(C(C)(C)C#N)=O)CCC12CCCN(C(c1cnnc(O)c1)=O)C2 C1(C(N2CC(C(C)NC(=O)Cc3cc(C4CC4)no3)C2)=O)CCc2c[nH]nc2C1 c1(Oc2cc(OCc3cc(C(=O)OC)c(C)o3)ncc2)cc(F)cc(Cl)c1 C(=O)(C1=NOC(c2ccccc2)C1)N(CCCCNC(=O)CC1CCCSC1)C C1(C(=O)NC(CN(C(C2(CC)CCCC2)=O)C)(C)C)C2C(=O)OCC12Br C1(Nc2nccc(SC)n2)CC2CC(C1)N(C(C1(CO)CCCO1)=O)C2 c1(C(N2C(CCNC(C(C)NC(CC)=O)=O)COCC2)=O)cc(F)c(F)cc1Cl C(c1ccn(C)c1)=CC(=O)N(CCN(C(c1c(SC)ccs1)=O)C)C C1(NC(c2cc(Br)c[nH]c2=O)=O)CCN2CCCC2C1 N1(C(c2n(C)ncn2)=O)CCC2(CC(NC(c3cnn(C(F)F)c3)=O)C2)C1 CCCCC(C(=O)N1CCCC1(C)CNC(=O)C(C#N)C1CC1)NC(N)=O C=C(CNC(=O)CNC(=O)CNC(=O)CC1(COC)CC1)c1ccccc1 S(=O)(=O)(c1cnccc1N1CC2CC2C1)N1CC(C)(C)OCCC1 N1(C(C2C(CC)C2)=O)CC2CCCC(C1)N2c1ncc2c(n1)COC2 C1(NC(=O)CN2CCN(CCc3ccsc3)CC2)CCc2c[nH]nc2C1 c1(C(N(CC(C)NC(C2CCC(=O)N(C)C2)=O)CC)=O)cnc2c(C)nsc2c1 CC1CCN(c2nccnc2F)CC1NC(=O)C(Cc1ccsc1)NC=O c1(C(=O)NCCc2ccn(CC)n2)cc(F)c(F)cc1Cl Cc1coc2c(CC(=O)NC3CC(C)CN(C(=O)C(O)C(F)(F)F)C3)cccc12 Cc1ccc(C(=O)NCC2(C)CCCN(C(C3CC(=O)N(C)C3)=O)C2)c(O)n1 c1(SC(C)C(=O)NCC(CO)NC(c2cnc(O)s2)=O)ccccc1Cl N1(C(=O)CN2CCOCC2=O)CC2CCN(C(c3ccc4nsnc4c3)=O)C2C1 C1(COC)CCCN(C(C2CN(C(=O)CC3CC=CC3)CC2F)=O)C1 c1(CCC)cccc(C(=O)NOCC(=O)N(n2cc(C3CCOC3)nn2)C)c1 n1(CC)nc(C(=O)NC(CC(=O)N2CCCC2)c2cccs2)c2ccccc12 C(C(C)(O)CNC(C1CC(CNC(=O)CCNC(=O)CO)C1)=O)SC c1(NC(=O)NC(c2ccc(F)cc2)C(C)C)c(Cl)cnn(C)c1=O CS(=O)(=O)c1cc(C(N2CCC(NC(=O)Cc3c[nH]c4ncccc34)C2)=O)co1 N1(C(C2C(=C)C2)=O)CC2COCCC2(NC(c2cn(CC(F)(F)F)nn2)=O)C1 N1(C(c2scc(C#N)c2)=O)CCOC2(CCN(C(c3ncncc3Cl)=O)CC2)C1 c1(C(=O)NC2CN(Cc3cc(F)cc(Cl)c3)CC2F)csc2c1CCCC2 C1(NC(C(C)SC)=O)CN(C(=O)C=CSCc2ccco2)CC1C C12(CNC(C(C)=C(CC)C)=O)CC1CN(C(c1cnn(CC)c1C1CC1)=O)C2 c1(C(=O)NC(C(C)NC(c2cnc(CC)s2)=O)C)cc2ncccc2o1 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(O)C3CC3)CC2)c2ccccc2n1 CC1CN(CC(N)=O)CCN1c1cc(NC2(C3CCCO3)CC2)ncn1 N1(C(CC=C)=O)CCCC2(CCN(C(=O)CC3CCC4CC4C3)C2)C1 N1(C(CC)=O)CCCCC(CNC(c2cn(-c3ccccc3)c(C)n2)=O)C1 c1(C(=O)NC(C)CNC(=O)C(c2cncc(F)c2)C)cc(C(F)F)cc(F)c1 c1(C(N2CC(F)CC(NC(=O)CC(F)(F)F)C2)=O)cccc2cnccc12 S(=O)(=O)(c1cccc(F)c1F)NCC(=O)NC(CC(N)=O)C(=O)O C1(NC(CC2OCC(C)(C)C2)=O)CC2CC1CN(C(c1ccccc1Cl)=O)C2 c1(C(=O)NCC(C2CC2)NC(CCCOC(C)=O)=O)nc2cccnc2s1 c1(OC)ccc(S(=O)(=O)N2CC3(CC(C(=O)Nc4ncc(C#C)cc4Cl)C3)C2)cn1 C1(C(=O)NC(C2CCOC2=O)(C)C)CCCN(C(C2CC2(F)F)=O)CC1 S(=O)(=O)(c1ccc(C(=O)O)cc1)N1CCC(NC(c2ccc(C)nc2)=O)C1 N1(C(Cc2cccc(-c3c(C)cc(OC)nc3)n2)=O)CCC2(CCCO2)C1 C(=O)(C1CCCc2n[nH]cc21)N1CCOCC(NC(CCC(C(C)(C)C)O)=O)C1 c1(CC)ccc(C)c(C(N2CCN(C(=O)Cc3cccc(F)c3)C3CC23)=O)c1 CCC(C)CC(=O)NC1C2CC1N(C(=O)C(C1CCCO1)OC)C2 C1(NC(=O)CC2(c3ccccc3)CC2)CCCC1NC(c1sccc1C(F)F)=O c1(CC(N2CCC(CCNC(CCC=C)=O)CC2)=O)ccc2c(c1)CCN2C c1(C(N2CCC(NC(c3ccc(COC)s3)=O)C2C)=O)ccc(F)c(F)c1 C1(C(N(CCNC(c2ccc(OCCC)cc2)=O)CCC)=O)CC2(C1)CC21CC1 CC1=C(C(=O)NCCCNC(=O)C(C(C)C)N2CCCS2(=O)=O)CCC1 C12(C(=O)NC(CNC(c3cn(CC)nc3C)=O)C3CCC3)CCC(N=[N+]=[N-])C1C2 CC(C)C(CNC(c1ccc(NC(C2(CN(C)C)CC2)=O)o1)=O)OC(F)F N1(C(=O)C(F)C2CCOC2)CC(F)(F)c2ccccc21 c1(C(N2CCC(F)(F)C(NC(=O)C(F)(F)C(F)F)C2)=O)coc2cc(O)ccc12 c1(C(N2CCC(NC(Cc3c(C)noc3)=O)(CF)C2)=O)cc(=O)n2ccsc2n1 c1(C(=O)NC2CC3CC(NC(CCCCSC)=O)C3C2)cn2ncccc2n1 C1(NC(C(C)NC(C)=O)=O)CCC(NC(=O)C(F)CC2CC2)CC1 N1(C(CCC#C)=O)CCC2(CC1)CCN(C(c1cc(OCC)ncn1)=O)CC2C Cc1cc(F)c(C(N2CCOC3(CCC3)C2)C(=O)NC2CCOC2)nc1Br c1(CC(C(=O)N(CC(C)NC(=O)CSC2CC2)CC)C)c(C)nn(C)c1C N1(C(CC)C)CC(C(N2CCN(C(=O)CSCc3ccccc3)CC2)=O)CC1=O CCC(C)CC(C(=O)NCC(C)COC)NC(=O)CCN1CCCCC1 C(C)(C)(C(=O)NC1CC(CCNC(C2CC2c2cccnc2)=O)C1)OCC C1(C(N2CC(NC(c3c(CC)c[nH]c3)=O)C(C)C2)=O)Cc2ccc(F)cc2C(=O)O1 N1(C(C(C)N(C)C)=O)CCC(C(=O)C(C)(C)C)CC1 CC1(C)CCC(F)(F)CC1C(=O)NCC1(CNC(=O)CN2C(=O)CNC2=O)CC1 CC1CCC(C)(C(N2CC(C)(NC(=O)CC(C)(F)F)C2)=O)C1 C1(CC=C)(NC(=O)CCCCCC)CC2CCC(C1)N2C(=O)Cc1n[nH]c(=N)s1 c1(NC(=O)NCCCN2CCN(Cc3n(C)ccn3)CC2)cccc(F)c1F C(C(CC(=O)N1CC(O)(n2ccnn2)C1)OC)NC(C(CC)C1CCCO1)=O N#CC1(C(=O)NC2CCCCC2CNC(=O)CC(F)(F)F)CC2CCC1CC2 CC1(C(=O)NC2CC(CNC(=O)Cc3cncs3)C2(C)C)CCOCC1 C1(NC(c2cc3c([nH]2)CCCC3)=O)C2CC3CN(C(=O)CCCCCF)C1C3C2 C1(CCNC(C2C(C(=O)OCC)C2)=O)CCCCN1C(=O)CCC1CC(F)(F)C1 CCC(C)(C(=O)NCCCCc1cn(-c2ccn(C)n2)nn1)NC(C)=O C1(CCC#C)CCCN(c2ccnc(NC3CCOC3)n2)C1 C1(N(CCO)Cn2ccc(C(CC)CC)n2)CCCN(CCCO)C1 c1(C(C(N2CCC(C(C)Nc3oc(C)cc3C)C2)=O)N(C)C)ccc(F)cc1 Cn1cc(C2CC2C(=O)NCCCn2cc(CNc3cscn3)nn2)nn1 Cc1cc(C(=O)NCC(CO)NC(c2csc([N+](=O)[O-])c2)=O)c2cnccc2c1 c1(CCC)c(C(=O)NCCCN(CCO)C(C2CC3(CCC3)C2)=O)nnn1C C1(C)(C(N(CCCCNC(c2c[nH]c(C(N)=O)c2)=O)C)=O)CCCCNC1=O N1(C(C(CCCC)O)=O)CC2CCC(C1)N2C(C1(C)CC2CCC(C1)S2)=O N1(C(C(C)NC(=O)NC)=O)CCC(NC(c2cc(Cl)ccc2O)=O)C(C)(C)C1 C1(C)CCC2(CCC2)OC1.c12ccc(cc1)CNC2C(F)(F)F.OC Cc1ccc(I)c(C)c1NC(=O)C(C1CCN(Cc2ccc(I)o2)CC1)C CN1CCN(C(=O)C(C2CCCCCCC2)O)CC(O)C1 C(=O)(C(C)CCC(C)(C)C)NCC(CC(=O)N(CC(CCCC)CC)C)C CC1CN(C(c2cccc[n+]2[O-])=O)CC1N(C(=O)C(F)(F)Oc1ccccc1)CC c1(C(=O)NCC(CNC(C2(CC#C)CCCC2)=O)(C)OC)[nH]nc([N+](=O)[O-])c1Cl CC1(C)C(NC(=O)C=Cc2ccncc2)CCN1c1ncc(C(C)(C)O)cn1 N1(C(=O)C2=NOCC2)C2CCC1(c1nn[nH]n1)CC2 C12CC(F)CN(C1)C2=O.c1(NC(=O)CN2CCCC2CO)cc(Cl)ccc1O c1(C(=O)NC2CC(NC(C3(COCC)CC3)=O)C2)ncc(P(C)(C)=O)cn1 c1(CC)cc(OC)ccc1C(N1CC(OC)C(NC(=O)CC2(O)CCC2)C1)=O c1(C(=O)NC2(C#C)CC2)conc1CNC(c1ccn(C)c1)=O C(=O)(C1CCCc2nccn21)NC1C2CCN(C(c3cc(OC)c(Cl)cc3)=O)C21 N1(c2cc(C)ncn2)CC(C)(C)c2ccccc21.C1CC(C)CC(C)(C)C1 N1(C(CC2(OCC)CCC2)=O)CC(CC(=O)NCC(F)CO)CC1(C)C C(=O)(C#CC(C)(C)CNC(C1CC1CCOC)=O)NCC(CC)(C)OC c1(NC(c2ccc(C(F)(F)F)s2)=O)cc(C2CCCCC2)nc2c(Cl)cccc12 C12(C3C(C)OC(C)C3)CC1COC2(C)C.C1CNCCO1 c1(SC(C(=O)NCCC(CNC(CNC(CC)=O)=O)O)C)ccc(C)c(C)c1 C1(C(N2CCC(O)(CN(C(CC(C)C3CC3)=O)C)CC2)=O)OC(C)(C)OC1(C)C Cc1noc(CC(=O)NCCCC(C)NC(C2CCC(=O)N2)=O)n1 CC1=C(C(=O)NC2C3CCN(C(c4nn(C(F)F)cc4Cl)=O)C23)SCCO1 C1(C)(C(=O)NCC2(C)N(C(c3cc(OCC)n[nH]3)=O)CCC2)CCN(C)CC1 C1(c2nnnn2C2CC2)(CNCC(CCC)OC)CC2CC2C1 c1(C(=O)N=c2[nH]nc(C3CCCOC3)s2)ccc2c(c1)OCCNC2=O CCC(C)C(O)CC(=O)NC1CCOC1C(=O)NC(C)C(=O)N(C)OC c1(C(N(CCCN(C(=O)Cn2[nH]cnc2=N)C)C)=O)nn(C)cc1Cl C12(C(=O)NCCc3ccc(Cl)cc3)CC1CN(C(C1C=CCN1)=O)C2 C(C1c2ccsc2CCN1C(=O)CSc1cn[nH]c1)NC(=O)Cn1nccn1 N1(C(c2c(C)cncc2)=O)CCN(C(c2cn3cccnc3n2)=O)CC(C)C1 N1(C(Cc2ccc(C)o2)=O)CCC(O)(CNC(=O)CCOCC2CC2)CC1 c1(C(=O)NCC(CO)NC(c2c(CC)nc(C)o2)=O)ccnc2cc(C)ccc12 C1(C(=O)NCC2CC(C(=O)NCCOCCOC)C2)CC2C=CC1O2 c1(C(C)NCCNC(=O)N(CCF)C2CC2)nnnn1C1(C)CC1 c12ncc(F)c(n1)C1(CCC1)N2.C(CC)(C(=O)N(CCO)CC)OCC c1(CC)ccc(C(=O)NCC2CCCC2NC(=O)CC(C)(F)F)c(F)c1 C(=O)(C(F)(CC)C(=O)OC)NCCN(C(c1ccc(CC)o1)=O)C1CC1 N1(C(c2c(CNC(=O)Cc3ccc(F)c(O)c3)noc2)=O)CCC12CCCSC2 C=CC1(CCNc2ccccc2CC(F)F)CCCCC1 C1(CNC(c2c(C)n[nH]c2)=O)COC(C)(C)CN1C(c1cnn2cnnc2c1)=O O=[N+]([O-])c1ccc(=NCc2cccc3occc23)[nH]n1 N1(C(CC(C)C)=O)CC2CCCCC2(C(=O)CCC(C)(F)F)C1 N1(C(C(C)C)=O)CCCCC1C(N1CCC(O)(CNC(C2CC3CC2C3)=O)C1)=O C(CO)(C(C)N=c1nc(N(C)Cc2cccc(C)n2)c2c([nH]1)CSC2)SC N1(C(C(=O)Nc2c(CN)scc2)=O)CC2(CCCC2N)C1 c1(OC(C)C)cccc(C(=O)NC2C3CC2N(C(c2nccn2C)=O)C3)c1 C(=O)(C#Cc1ccccc1C#N)N1C(C)CC(NC(c2cn(C)c(=O)n2C)=O)C1 N1(C(c2cocc2Br)C(=O)NCCSC)CCN(C)c2ccccc2C1 N1(C(C2C(CCC)C2)=O)CCCCCC1C(N1CC(CO)C(CO)C1)=O C1(C(=O)NC2C(CCOC)CCC2)CC(N=[N+]=[N-])CN1C(c1nnn(C)c1C)=O c1(OC)cc(CN(CC(O)CN(C(=O)C(=O)NC(C)C)C)C)cc2c1OCCO2 c1(C(=O)NCC(C(C)C)NC(C(c2scc(C)n2)(F)F)=O)cnc2cccnn12 c1(NC(c2cc(-c3cccc4c[nH]nc34)cnc2Cl)=O)ccc([N+](=O)[O-])cc1F N1(C(C(C2CC2)SC)=O)CC2CC1C2C(=O)NCCC1CCCC(C)C1 CC1OC2(C)CC1(C(=O)NCCN(C(=O)C(O)C(F)(F)F)C1CCCCC1)C2 C1(CCC(=O)NC(C)CCN(C)C)CCN(C(C2(C#N)CC2(C)C)=O)CC1 c1(C(N2CCC3C2CCN3C(C2CC=CC2)=O)=O)ccc2ocnc2n1 CCC(C)C(C(=O)NCCN(C(c1cn(CC2CCCCC2)nn1)=O)CC)OC Cc1ccc2c(c1)SC(C(=O)NC1CC1NC(=O)C(C)(C)c1nncn1C)C2 C=CCC(C(=O)NCC(C1CC1)N(C(=O)CCN(S(C)(=O)=O)C)C)C(C)C c1(OC)cc(NC23CCC(NC(=O)C(C)(C)C)(CC2)C3)ccc1[N+](=O)[O-] c1(C(=O)Nc2cncc(F)c2)ccc(SC(Cc2ccccc2)CO)cc1 CC1(CC(N)=O)CCN(C(=O)CC2CCN(C(=O)CCC3CCOCC3)C2)CC1 C1(C(N2CCC(C)(NC(C3C(CC)OCCC3)=O)C2)=O)CN2CCC1CC2 C12(C(N3C(CN(C)C(c4ccc5c(c4)CC5)=O)CCCC3)=O)COC(CCO1)C2 C1(NC(=O)Cc2cccnc2)CC2CCC(C1)N2C(c1nc(O)nc(O)c1F)=O C1(NC(c2ccc(F)cc2F)=O)CC(O)CN(C(c2[nH]cc3c2CCC3)=O)C1 C1(C(=O)NC(C)CCNC(=O)Cc2cncnc2)CN(C)CC1C(F)(F)F c1(C(N2CCC(N(C(CCOCC)=O)C)C2)=O)ccnc2ncc(C)cc12 c1(CNC(C)=O)cc([N+](=O)[O-])ccc1N1CCN(C(=O)C=Cc2cscn2)CC1 Cc1[nH]nc2ncc(C(=O)NC3CCC(C)N(C(=O)CCC4CC4(F)F)C3)cc12 c1(C(=O)NC2CC(OC)CN(C(c3cc(CC)no3)=O)C2)c(C)cc(C)cc1Cl c1(C(=O)NCCC2(NC(C3CC3Cl)=O)CCOCC2)c[nH]cc(Cl)c1=O c1(C(=O)NCCC(C)N(C(=O)CC2COC(=O)C2)C)ccc2c(c1)CCO2 C(C)(C(=O)NC1CC2CCC1N2C(c1csc([N+](=O)[O-])c1)=O)(C(C)C)OC C1(NC(c2[nH]cc(C(C)(C)C)c2)=O)CCCCN(C(C2CC(=O)C2)=O)C1 C(CN=c1[nH]c(=NC2COCCOC2)[nH]c2c1SCC2)(c1ccoc1)OC C1(NC(CN(C2CC2)CC)=O)CCC(C)N(C(c2cn(CCO)nn2)=O)C1 N1(CC)CC(C(=O)NC2CCCC(NC(=O)CCc3cnc[nH]3)C2)CCC1=O N1(C(C(C)(C)SC)=O)Cc2[nH]nc(C(=O)NCc3cc(C)co3)c2C1 Cc1csc2ncnc(N(C(C3CCCNC3)C)Cc3c(Cl)ccc(Cl)c3F)c12 Cc1ccn2cc(C(N3CCC(C)(C)C3CNC(C3CC4CC4C3)=O)=O)nc2c1 CC(N=c1cc[nH]cc1S(=O)(=O)N(C1(C(N)=O)CCC1)C)C1CN(C)CCO1 N1(C(C(CC)N(C)C)=O)CCN(C(c2scc(C)c2Br)=O)C(C)C1 C1(CCN(C)C(c2cscc2C(N)=O)=O)CCN(C(=O)C2=NOCC2)CC1 C1(C(N2C(C#C)CCC2)=O)CN(C(C2CC(=O)N(CC)C2)=O)CC1(C)C N1(C(C=C(CCC)CCC)=O)CCN(C(C2CCC(C(N)=O)O2)=O)CC1C C=C=CCC(=O)N(CC(C)(C)CNC(C1CCCOC1)=O)C C1(NC(CCc2n(C)cnn2)=O)C=CCC(C(N2CCC(C)(F)C2)=O)C1 N1(C(c2cccc(C)c2N)=O)CCC2(C1)CN(C(C1(C)CC1(Cl)Cl)=O)CCO2 C(=O)(C(C)(F)C(=O)NCC1CC12CCCCC2)OCC.C12CCN(CC1O)C2=O CC(C(=O)NCc1cccnc1NC(=O)C(Cc1cnc[nH]1)N(C)C)S(C)(=O)=O C(C(C(=O)N(CC(C)N(C(=O)C1=CCC1)C)C)OC(C(C)(C)C)=O)OC C1(N(C(c2c(CC)onc2)=O)C)CN(C(=O)Cn2cc(C)cn2)CCC1C c1(C(=O)NCC2CC3CN(C(c4csc(C)c4C)=O)CC32)c[nH]c2nccc-2c1 C(CCCCC(=O)NCC1CCCCC1NC(C12CC(C(C)(C)C)(C1)C2)=O)OC C(C)(N=c1[nH]c(=N)[nH]c(=NC(CCc2ccccc2)C(C)C)[nH]1)c1c(CC)nns1 C12(C(=O)NCC3N(C(c4n(C)ccc4)=O)CCCC3)CCOC1CC(=O)NC2 N1(C(CC(=C)Br)=O)CC(NC(=O)CN2C(=O)CN(C)C2=O)CC(C)C1 N1(C(C2(OC)CCCOC2)=O)CC(C(=O)NCC2CC2C(C)C)CC(C)C1 N1(c2c(OC)nc(Cl)nc2)CCC2(CCC(F)(F)CC2)C1 N1(C(C2(C3CCC3)C(C)C2)=O)CC2CCC1CN2C(=O)C1CC1 N1(C(CC(COC)(C)C)=O)CC2(C)CC1(C(=O)NCC=CCSC)C2 C=CC1(C(N2CC3C(N(C)C(c4cccc(C)c4Cl)=O)C3C2)=O)CCCCC1 n1(CC)c(SCC(N2CCCC2)=O)nc2ccccc12.S1(=O)(=O)C2CC(C2)N1 C(C(C(=O)NC1CCOCC1C)C(C)C)NC(CCCC=C)=O c1(C(C(=O)NC2C(CNC(c3cn(CCOC)nc3)=O)C2)F)ccc(F)cc1 CC(C(C)C)=CC(=O)NC(C)(C)CN(C(=O)CCC1CC1(C)C)C c1(NCCN2CCN(C(COC)C)CC2)nc(C)ccc1OC c1(Nc2nc([SH](c3c(F)cccc3Cl)C(C)=O)c(Br)s2)cc2c[nH]nc2cc1Cl Cc1cnc(N2CCC(c3ccc(C)c(C)c3)C2)nc1C.N12CC(O)CC1C2=O c1(C(N2CC(CC)N(C(=O)CC3CCCC(C)O3)CC2)=O)cc2cccnn2c1 N1CCS(=N)(=O)C2(CCC2)C1.Cn1ncc2cccc(N)c12 Cc1ncc(Cl)c(C(=O)NC2CN(C(=O)C3=CCCOC3)CC2C(F)F)n1 Cc1sc(N)c(C(N2CC(NC(=O)C(C)c3cccs3)CC(C)C2)=O)c1C c1(CC(=O)NC2(CNC(=O)CCSc3cn[nH]c3)CCC2)ccc([N+](=O)[O-])cc1 CC1(C)COC(=O)C1NC(=O)CCCn1cc(CC2CCCOC2)nn1 c1(C(N(CCCNC(c2c(C)nc(C3CC3)o2)=O)C2CC2)=O)cncc(C#N)c1 c1(C(=O)NCC2(OC)CN(C(C(C)NS(CC)(=O)=O)=O)C2)ccccc1CO C=C(C)CCC(C)NC(C1CCC(NC(=O)CC2CC(=O)C2)C1)=O Cc1ccc(C)c(C(=O)NC2COCCN(C(=O)C(c3ccc(O)cc3)=O)C2)n1 N1(C(c2c(C)n(C)cn2)=O)CC(C(N2CCC3CC23C)=O)CC(C)C1 Cc1cccc(C(=O)NC2CC(C(C)NC(c3cn(C(C)C)nc3C)=O)C2)c1C c1(N2C(C)CC(CNC(C3(C)C=CCC3)=O)C2)cc(C#N)ccc1[N+](=O)[O-] N1(C(c2c(C)nc(CC)o2)=O)C2CC=C(C(=O)NCC3CC3C(=O)NC)C1CC2 N1(C(c2c(C)nn(C)c2)=O)Cc2ccccc2C(CNC(C2CC2C(C)O)=O)C1 Cc1cccc(CC(=O)NC2CCCC(NC(c3cc(C)oc3C)=O)C2)c1 c1(COC)ccc(NC(C2(NC(c3occc3C)=O)CCCC2C)=O)cc1 N1(C(COCC(=O)NC)=O)CC2CCC2(CCNC(c2cnc(C)cc2Cl)=O)C1 c1(CN=C(NCc2cc(C)on2)NCC(C)(C)C(C)(F)F)noc2c1CCCC2 CCCC(CNC(C1CC1[N+](=O)[O-])=O)C(=O)NCC(=O)NOCC Cc1ccnc(C(N2CCN(C(=O)C(C)SCC3CCCO3)CC2C)=O)c1O C(=O)(C1=C(C)CCCC1)N1CC(CC=C)(NC(C2CCOC2C(F)(F)F)=O)C1 N1(C(c2cc(Cl)cc(Cl)c2Br)C(=O)NCC(=C)C)CC2(C)CCC2(C)C1 N1(C(Cc2cncc(C#N)c2)=O)C2CCC1C(F)C(NC(c1nsnc1O)=O)C2 C#CCCCCC(=O)NC1CCCC1(C)NC(=O)C(c1ccccc1)C Cc1c(C(N2CCN(C(c3ncn(C)n3)=O)CC2C)=O)ccc2c1CCC2 N1(C(c2cccc(CNC(COC(C)=O)=O)n2)=O)CCCC(CO)CC1 c1(OC)ccc(C=CC(=O)NCCNC(c2c(Cl)c([N+](=O)[O-])nn2C)=O)c(C)c1 N1(C(CCC(C(C)C)NC(=O)CCC2CCCO2)=O)CCCC12CCOCC2 c1(NC(=O)OC(C)(C)C)ccsc1NC(=O)NCc1ncc(Cl)s1 c1(CC)ccc(CN(C(=O)C(c2ccco2)NC(c2cc(C)co2)=O)C)o1 C1(C(=O)OC)CCCCC1C(=O)Nc1nc(-c2ccccc2C(=O)NC2CC2)cs1 C1(CNC(C(CC)NC(N)=O)=O)CCN(C(=O)CC2CCC(=O)N2)C1(C)C C1(C(=O)Nc2ccc(OC)cc2)CN(C(=O)CCCn2ccnc2)CCC1(F)F C1(C(N2CCC(C)N(C(C3CC4CCC3O4)=O)CC2)=O)CCc2ccccc2C1 C(=O)(N=c1[nH]c(Cl)ncc1O)C1CCCN(C(c2c(C)nc(Cl)cc2)=O)CC1 N1(C(C(C)OC(C)C)=O)CCC2(CCN(C(c3cc4c(s3)CCOC4)=O)C2)C1 C1(CC)CNC(=O)CN1C(=O)C(C1CC1)N(C(=O)CNC(=O)OCC1CC1C)C c1(N(C)C(=S)NC(=O)CC2=NNC(=O)C2)c(Br)cncc1[N+](=O)[O-].C1COC1=O C1(OC)CN2CCCC2(C(N2CCOC(CNC(C3CC3(C)C)=O)C2)=O)C1 C1(C(N2CC(NC(CC(CC)OC)=O)CC2(C)C)=O)CC(C)(C)OC(C)(C)C1 Cc1noc(C)c1CN1CC2C(C(=O)NCCCC3CCOCC3)C2C1 c1(C(N2C(C(C)(C)NC(c3cnns3)=O)CCC2)=O)cc2cc(Cl)ccn2n1 C1(C(=O)NC2CC(CCNC(c3ccn(CCC)n3)=O)C2)CC(=O)N(C)C1 N1(C(c2ccc(CSCC)cc2)=O)CC2CC1CN2C(C1CC(C)=NO1)=O C1(CNC(C2CC3CCC2O3)=O)CN(C(c2ncc(C(F)(F)F)s2)=O)CCO1 C1(NC(Cc2c(C)n[nH]c2C)=O)CC=C(C(=O)NC2CC2OC(F)F)C1 CC(CNC(C1CN(C(N)=O)C1)=O)C(=O)NCC1CCC1 CC1CCN(CCC(=O)NC2CCCC(N(C(=O)C=CBr)C)C2)CC1 c1(C(=O)NCCCCC2CN(CC=Cc3ncc[nH]3)C2)ccc(-c2ccsc2)cc1 CC1(C)CCOC1CC(=O)NCCC1CCCN1C(c1cnnn1C1CC1)=O C(=O)(CC1=NN(C)C(=O)C1)NC1CC(C(NOCCN(C)C)=O)C12CCC2 c1(C(N2CCN(c3ccc(C45COCC(C4)C5)s3)CC2)CO)cc(F)ccc1F c1(CC(CO)NC(c2n(C)nc(C3CCCO3)c2)=O)cc(Br)ccc1F c1(CNC(C=CC)=O)cc(C(=O)NC2(CCCc3ccccn3)CCC2)n(C)n1 c1(COC)nc(C(=O)OCC2(COC)CC2)c(-c2ccccc2)s1 c1(CCC(N2C(CC=C)CCC2)=O)nnc(S)n1C N1(C(=O)CN2CCOCC2=O)CC2CC(C1)CN(C(C1CCCS1)=O)C2 CC(C(=O)NCC(c1ccccc1)CNC(=O)CCC(=O)c1ccc[nH]1)C(F)F N1(C(CCOC(C)C)=O)CC(NC(=O)Cn2cnc(C(N)=O)n2)C(C)(C)C1 C1(C(=O)NC2CCC(NC(C(CC)(C)OC)=O)CC2)COCC(C)(C)O1 N1(C(C2CCC(C)O2)=O)CC(C)(C)CC1CNC(=O)CCC1CCCOC1 N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3CCC(F)CC3)=O)C2)C1 c1(C(=O)Nc2ccc(C(=O)Nc3ccc(F)c(Cl)c3)c(F)c2)c(Cl)cccc1Br N1(C(C2C(C)C2)=O)CC(N(c2sccc2Cl)C(=O)C(c2cncn2C)O)C(O)C1 Nc1ccc(Cl)cc1C(=O)NC1(c2cn(Cc3nccs3)nn2)CCC1 c1(C(=O)NCC2C(NC(COCCOCC)=O)C2)cc(OC)c2occc2c1 CC1CCOC1C(=O)NC1COCC1CNC(=O)CC1CCC1 c1(CC)ccc(C(=O)NCC2(CNC(C3CCCC3C(F)F)=O)CC2)cc1F N1(C(CC(=C)CN(C)C)=O)CCC2(CC1)CC(NC(=O)CC(O)CCC)CCO2 c1(C(N2CCC(NC(CCC(C)SC)=O)CC2C)=O)cccc2nsnc12 C1(C(=O)NCC(=C)CCNC(c2csc(-c3ncccn3)n2)=O)CCC(=O)NC1 c1(CCNC(=O)NC2CC3CN(C(=O)OC(C)(C)C)C2C3)nc2ncccn2n1 Cn1nncc1CC(=O)NCC1COCC1NC(c1scnc1Cl)=O c1(CN2CCCC(CC(=O)Nc3cnnc(Cl)c3)C2)ccc(O)c(O)c1 c1(C(N2CCC(F)(C(N)=O)CC2)=O)csc2c1CCN(S(=O)(=O)CCCCl)C2 N1(C(=O)COCC2CCCO2)CC2=C(C1)CN(C(c1cccc(O)n1)=O)C2 C=CCC(CNC(C1C2CCCCCC12)=O)C(=O)NCC1CC(OC2CC2)C1 c1(N(C(C)CNC(C2CCN(C)C2)=O)CC)nnc2c(c1C(=O)OC)CCC2 C(C(=O)NCCCNC(=O)C(C)(C)c1ccnn1C)(C(C)C)OC(C)=O c1(C(=O)NCC(C(C)C)NC(CN2CCCC(CC)C2)=O)ccc2cnoc2c1 c1(C(=O)NCCCOCCNC(C(C2CCCOC2)OC)=O)nc(O)c(C)s1 CCC(C)CCC(=O)N(C1CN(C(c2cc(Br)cnc2O)=O)CC1(C)C)C c1(C(=O)NC(C2(O)CCN(C(C=CCOC)=O)CC2)C)cc2scc(C)c2[nH]1 N1(C(c2c(C)n(C)nc2)=O)CCC2CN(C(c3cnn(C(C)C)c3N)=O)CC12 Cc1cnn(C)c1C1CCN(C(=O)NC2CC3CCC3C2)C1 c1(NC2C(C)CN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2C)nc2ccc(Br)cc2s1 C1(C(=O)NC2CCCCC2NC(=O)COCc2nccn2C)(OC)CS(=O)(=O)C1 C1(C(N2CCCC(C(=O)NC3CC(C)(C(N)=O)C3)C2)=O)CCOC(=O)CC1 C=CCC(C(=O)NC1CC(NC(c2cc(Cl)c(F)cc2F)=O)C(O)C1)C(C)C Cn1nc(C(N2CC3CC2CCN3C(=O)CC23CCCC2C3)=O)c2c1CCC2 c1(C(=O)NCCC2(NC(C=CC(=O)OCC)=O)CCC2)scc2c1OCCO2 n1(CC)nc(C(N2CCC(C(C)(C)NC(=O)CC3CCCCC3O)C2)=O)cc1O C1(C(=O)NCc2ncc(CC)o2)CCCCC1(C)NC(=O)Cc1csc(C)n1 Nc1cncc(C(=O)NCC(C2CCCCC2)NC(c2csnc2Br)=O)c1 c1(C(=O)NC2C(C=C)CN(C(C3(O)COC3)=O)C2)cc(Br)cc2c1OCO2 CC(C)C(O)C(C)C(=O)NCC1(F)CCCN(C(c2ccc(CO)nc2)=O)C1 CCCC(C(=O)N(CCCCN(C(=O)Cc1ccnn1C1CCC1)C)C)N(C)C c1(OC)ccnc(N2CC(O)(C(C)NC(=O)CC3(CSC)CC3)C2)n1 N1(C(COCC(=O)OC)=O)CC2CC(C(N3CC(O)(C(N)=O)C3)=O)C(C2)C1 N1(C(C(C)N2CCC2)=O)CCCC(n2cc(CNC(c3cccnc3)=O)nn2)C1 C1(CC(=O)NC(C)CC(N)=O)CC2(CC2)CN1C(=O)C(O)CC1CCCC1 C1(NC(c2scc(CNC(C(C)OCOC)=O)c2)=O)CCCCCC1(C)C CN1CCC(O)(CNC(=O)C(C2CCN(C(c3ccc(C(F)F)o3)=O)C2)F)C1 c1(C(N(C(C)CCNC(=O)Cc2nccs2)C)C)cc2ccccc2o1 C(=O)(CC(C)C(F)(F)F)NCC1(C)CCN(C(CC(C(C)C)O)=O)CC1 CN1CCOc2cc(CNC3C4CCC(C4)N3C(c3cn(C)cn3)=O)ccc21 Cc1nc(C(C)C)sc1C(N1CCOC(CCNC(=O)CC2COCC2O)C1)=O C(=O)(CC(C(=C)C)OCCOCC)N(C1(C(=O)OC)C(C=C)CC1)CCC N1(C(C(CC)C)=O)CC2CC1CCN2C(c1c[nH]nc1-c1ccncc1)=O c1(C(=O)NC2CCN(C(C3(CCC=C)CC3)=O)C2)cc2ncc(Br)cc2o1 c1(C(N(C)CC2CN(C(c3cc(OC)nn3C)=O)C2)=O)ccc2c(n1)CCC2 C12(NC(c3ccncn3)=O)CCC1CN(C(c1ccc(SC(F)(F)F)o1)=O)C2 c1(C(N(C2CCC(NC(c3c(N)cnn3C)=O)CC2)C)=O)cc2sccc2[nH]1 C(=O)(C(=O)NCC(=O)N(C)N(C)C)NC1CC(OC(C)C)C1.C12CC1C2 CCCC(F)(F)C(=O)NC(C)CN(C(=O)CNC(=O)OC(C)(C)C)C C1(NC(C(C)CC2CC2)=O)Cc2ccccc2C1NC(c1nc(O)[nH]c(=O)n1)=O c1(C(N2CC(n3cc(C(C)OCC)nn3)C2)=O)ccc(=O)n(CC(C)O)c1 c1(Nc2c(Br)ccnc2Cl)cc(Cl)ccc1[N+](=O)[O-].CC12CCCN1C(=O)C2 c1(N2CCC(CNC(c3c(OC)noc3C)=O)CC2)ccc(C)cc1[N+](=O)[O-] C1(C(=O)NC2(CC=CC(=O)Nc3cnc(O)c(F)c3)CCC2)CC2CCC1C2 C1(CNC2C(c3ccccc3)CCCC2)CCC2COCCC2C1 CC1(NC(C23CC2CNC3=O)=O)CCCCC1C(N1CC(C(N)=O)C2(CC2)C1)=O C(=O)(C1=NNC(=O)CC1)NCCN(C(C1Cc2cc(C)ccc2S1)=O)CC C#CCCC(C(=O)N1CCOC(C)CC1)NC(=O)Cc1cc(C)on1 C1(CN(C)C(c2cc[nH]c2)=O)CCN(C(C2CCC(CCO)CC2)=O)CC1 C(c1c(C)noc1C)=CC(=O)NCC(CNC(Cc1nc(C)c(C)[nH]1)=O)O C1(=CCNC(C(c2cccc(Cl)c2)C)=O)CCN(C(C2(F)CC=CC2)=O)CC1 Cc1c(C(=O)NCCC(C)NC(c2cccc(C(F)F)c2)=O)nn(C)c1Br Cc1cc(C(=O)NCc2cccc(-c3cn(CCF)nn3)c2)c(C)n1C1CC1 C(=O)(C1CC(C)(C)Oc2ccccc21)N1CC2C(CNC(C3(C=C)CC3)=O)(C2)C1 N1(C(C(CC)n2ccnc2)=O)CC(CO)C2(C1)CN(C(c1cc(N)cs1)=O)C2 c1(C(=O)OC)nnc(N2CCCC(CCCO)C2)n2ccnc12 N1(C(c2cn(CC)nn2)=O)CC2CCC1C(NC(=O)CNC(C)=O)C2 N1(C(c2cc(C)[nH]n2)=O)CCOCC(NC(c2ccc(C(N)=O)cn2)=O)C1 N1(C(C(C)N(C)C)=O)CCCC12CCCN(C(C1CC(C(F)(F)F)C1)=O)C2 c1(C(=O)NCCN(CCC#C)C)cc(CCC)[nH]n1 N1(C(c2c(C)onc2)=O)CCC(C2CCN(C(=O)C(O)CC[S+](C)C)C2)CC1 C(N=c1[nH]c(C2CC2(F)F)cs1)c1cc(COC)no1 C=CC(CCC)CC(=O)NC(CCC)C(=O)NCCC(=O)N(C)C Cc1ccc2[nH]c(C(=O)NC3CC4CCC3N4C(=O)Cc3ccns3)cc2c1C CC1(C)CCC(C(=O)NC(C(F)(F)F)C2CC2)CN1C(c1c[nH]c(=O)cn1)=O N1(C(C(C)OCC(F)(F)F)=O)CC(CNC(=O)CN(c2cncn2C)C)C(O)C1 C1(C(N(CC(C)O)C)=O)CC2CC1CN(C(c1coc(C(F)F)n1)=O)C2 N1(C(C2C(C)(C)C2(C)C)=O)C(C(=O)NC23CC(C2)C3)C2CC(O)C1C2 c1(CCC(=O)NC2C(NC(c3c(C(=O)OC)c[nH]n3)=O)C2)c(C)nn(C)c1C C1(C(=O)NCCn2cc(C(N3CCC(C)C3)=O)nn2)CC(C)(C)CO1 C(C(C)(C(=O)N(CCCn1ccnc1)CC(C)C)NC(c1ccncc1)=O)SC C1(O)(C(C)CNC(c2cn(C(F)F)cn2)=O)CCN(C(=O)CCc2cscn2)C1 C1(CNCc2cncc(Br)n2)CN2CCC1CC2 C1(NCC(=O)NC(CNC(c2c(C(C)(C)C)con2)=O)C2CC2)CCS(=O)(=O)C1 c1(C(=O)NC2C3CN(C(C(CC)(C)COC)=O)CC32)cc2cc(C)cc(C)c2[nH]1 CN1C(=O)CSC1=CC(=O)NCCCNC(c1cc(C#N)c(O)nc1N)=O C(=O)(N=c1[nH]nc(N2CCOCC2)s1)N1CC(C)SCC1 C1(C(N(C2CCCC2C#N)C)=O)(CO)CCN(C(C2CC(O)C2)=O)C1 CC(C)(C)CCC(=O)NC1CC1CNC(=O)CNC(=O)Nc1ccccc1Cl c1(C(=O)OCC)cnc(C)[nH]c1=NCC=CCNC(=O)C(C)S(N)(=O)=O c1(NC(c2n(C)nc(C3CC3)c2)=O)ccc(Br)cc1C1(C(=O)O)CCC1 c1(CCC(=O)N(CC(CC)NC(=O)CCNC(N)=O)CC)cc(C)no1 c1(C(N2CCN(C(=O)C3=CCCCC3)C3CCCC23)=O)cc(O)c2sccc2c1 CC1CC(NC(=O)Cc2cnccn2)CCN1C(c1ccc(F)nc1F)=O c1(C(=O)NCC23C(CN(C(c4c(C(C)C)ccs4)=O)C2)C3)ccnc(F)c1N c1(C(N)=O)nnc(CNC(c2nccnc2C(N)=O)=O)n1CCOCCO c1(OCC)ccc(C)nc1C(N1CC(C(C)NC(=O)Cc2ccc(Cl)nc2)C1)=O c1(CC)cccnc1C(=O)NC1(CNC(=O)CC(C)Cc2cccc(F)c2)CC1 C1(O)(CNC(CNC(CCC)=O)=O)CCN(C(C2(c3ccno3)CCC2)=O)C1 Cc1c(F)cc(-c2cnc(C(F)(F)F)cc2C(=O)NC(C)COC(F)F)cc1F N1(CC(=O)NC(c2n(CC)ncc2)C)CCN(C(=O)CCN2CCOC2=O)CC1 c1(CN(C2CCCCC2NC(c2cc(CC)c[nH]2)=O)C(CC)=O)ccccc1Cl C1(C)(CC)CC(NC(C2CN(C(c3ncccn3)=O)C(C)(C)C2)=O)CCO1 C1(CNC(c2ncc(C)nc2)=O)CC2CCC1N2C(=O)C(C1CCCCC1)F C1(C(=O)Nc2c(OC)ncnc2)CCN(C(c2ccc(F)s2)=O)CC1O C1(OC)CN(C(c2conc2C)=O)CC1NC(=O)C(=Cc1cnn(C)c1)C N1(C(C(C)(C)OCC)=O)CC(N(C(=O)CSc2ccc(F)cc2)C)C2(CC2)C1 C1(C(N(CCC)CCNC(=O)CC2CCOC2)=O)CCOC(C(C)C)C1 N1(C(=O)NC(C)C)CCC(C(=O)NCCCCN2CCC2)C(F)(F)C1 c1(OC)ccccc1C(C)C(=O)NCCCCNC(c1sccc1Cl)=O Cc1ccc(CCC(=O)NC2C=CC(CNC(=O)CC(=O)N(C)C)C2)s1 C1(C(=O)NC(CNC(C=CC(=O)NCCOC)=O)(C)C2CCC2)CCNC(=O)C1 N1(C(CCOC(C)C)=O)CC(C)(C)CC1CNC(C1CC1c1ccccn1)=O c1(C(N2CCCC2C(N(C2CC2)CC2CCCO2)=O)=O)cc2ccc(Cl)cc2[nH]1 c1(OC)ccc(C(N2CC(NC(C3CC3CC(C)(C)C)=O)C2)=O)c2ccncc12 C1(CNC(C2(OC)CCC2)=O)CC(C(=O)N2CCCCC2C)=NO1 c1(NCC2(C)CC(C)(C)C2)ccc(S(=O)(=O)N2CCCC(C(=O)N(C)C)C2)c(Br)c1 N1(C(C=C(C)C)=O)CCC2CC12C(=O)NC(c1nc(=O)o[nH]1)C c1(C(=O)NCC(CO)NC(c2csc(Cl)c2)=O)ccc(C2CC2(F)F)cc1 N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CN(C(=O)C1=CCCOCC1)CCO2 C(C)(C(C(C)C)NC(=O)CC1CC(F)(F)C1)NC(C=CCOCCOC)=O N1(C(c2[nH]cc(CC)c2)=O)CCC2CN(C(=O)COCCF)CCC12 C1(C(=O)NCCCCCN(C(C=C(COC)C)=O)C)CCCC(C(C)C)C1 N1(C(C2(C)CCCC2)=O)CC2CC(NC(c3cnn(CC(F)F)c3)=O)CC2C1 C1(NC(c2cc(OC)no2)=O)CC(NC(c2n[nH]c(C)c2Br)=O)CC1O c1(CCC(=O)N(CC(=O)NC(CC=C)C2CC2)C)cncn1C C1(CNC(c2n(CCC)ccc2)=O)CN(C(=O)C=Cc2cnc[nH]2)CC1O C1(CNC(c2cc(Cl)cc(Br)c2)(C)C)CCc2ccccc2O1 CCCCC(O)C(=O)N1CCOC(CCNC(=O)CC(C)(C)SC)C1 c1(CC(=O)NC2C(CNC(=O)C=CC3CCCO3)CCC2)csc2nccn12 C(=O)(CC1=CCN(C)CC1)NCCCC(C)NC(=O)C(F)CC1CCCC1 Cc1cccc(C)c1CNCC(O)C.N1(CC(C(=O)O)N)CCCS1(=O)=O c1(OC)nc(C(=O)NC(C)(CNC(C2CC2F)=O)C2CC2)sc1C C1(CCNC(CC2(C=C)CC2)=O)(NC(=O)C(F)(Cl)c2ccccc2)CCOCC1 c1(C(=O)NCC(C)NC(=O)OC)cc(CNC(C2CC3(CC3)C2)=O)cn1C C1(CC=C)(C(=O)NCC2CSC2)CCCN1C(c1cc(CCC)on1)=O c1(C(N2CC3C(C2)N3C(c2ccc(I)cc2Cl)=O)=O)ccc(F)c(F)c1F N1(C(c2ccnc(C)n2)=O)C2CCC1C1CC1(NC(=O)Cn1nnc(=O)[nH]1)C2 C(=O)(C1Cc2ccccc21)N1CC(NC(c2ccc(CCF)cc2)=O)C(O)C1 C(=O)(CC(C)(C)CNC(C1CC(O)C1)=O)N1CC(NC)C1 c1(C(=O)NC(C)CN(c2ncc(C#N)cc2Cl)C)ccc2c(n1)CCCN2 C1(C(=O)NCC2CCCO2)CC12CCN(C(c1cn(CC3CCC3)nn1)=O)CC2 Cc1cc(Cl)cc(C(N2CC(C3CN(C(=O)CCn4cccn4)C3)C2)=O)c1N C(=O)(C1=CC(O)C(NC(=O)CC(C)O)C1)N1C(CC(=O)OC)CCC1 c1(C(C)=O)cc2ccccc2cc1C=CC(=O)NC(C)CNC(=O)C(C)C(F)F n1(CCC(=O)NCC(C2CCC2)NC(C(C)NC(C)=O)=O)c(C)csc1=O Cc1ccnc2c(C(=O)NC3CC3CNC(=O)CN3CC(C)C3)cccc12 C(=O)(C1CCCc2cccnc21)N(C(CNC(C1OCCO1)=O)C1CC1)C c1(CC(C)C)nnc(C(=O)NC2CCN(C(=O)COCCOCCO)C2)s1 C1(C(N2CC(C)C(C)(CNC(c3cnncc3O)=O)C2)=O)Cc2ccccc2O1 c1(C(=O)NCC2(O)CN(C(CC3(C)CC3F)=O)C2)cccc(Cl)c1O c1(C(=O)NCC(CO)NC(=O)C(c2ccc(Cl)cc2)O)ccc(O)cc1C(F)F O=C(C1=NOC2(CCN(C(C3CC3(F)Cl)=O)C2)C1)NCc1ccc(F)cc1Cl c1(OC)ccc(NC(=O)NCC(CO)SC)cc1OC(F)F N1(C(C(C)Cn2ccnc2)=O)CCCC(C2CN(C(C3(C4CC4)CCC3)=O)C2)C1 N1(C(CC(CC)C2CC2)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC2(CC2)C1 C(C1=NOC2CN(C(c3ccnc(C)n3)=O)CC12)NC(C=C(COC)C)=O CCC(C)(COC)C(=O)NCC1(F)CC(CNC(=O)CC2CC(C(F)F)C2)C1 CCC(c1ccc(Cl)cc1)=CC(N1CC(OC)CC(CC)C1)=O C1(CCC(=O)N(CC(=O)N(C)C)C)CCN(C(C2CCC2(F)F)=O)CC1 C1(C(=O)NC(CN(C(C=CC)=O)C)(CO)CO)CN(S(N)(=O)=O)C1 C1(CC#C)(C(=O)NCc2cccnc2)CCCN(C(=O)CC(=O)OCC)C1 N1(C(C(C=C)(C)O)=O)CC2(C1)CN(C(=O)CNC=O)CCO2 C(C)(C(CC(=O)NC1(CO)CC(C)(C)C1)NC(=O)CCC(=O)NC)OC C(=O)(C(C)(C)C1CCCN1C(=O)Cn1cc(CO)nn1)N(CC(=C)C)CC CC1(C)C(C(=O)NCC(=O)NCC2CCN2C(=O)Cc2nccs2)C1(F)F C12(NC(c3c(C)cn(C)n3)=O)COC(C1)C(NC(c1cc(Cl)cs1)=O)C2 N1(SCC(COc2cccc(CC)c2)O)C(=O)NC2(CCCSC2)C1=O c1(C(=O)NC2C(NC(CC(CCC)(C)C)=O)CCC2)ccc(S(C)(=O)=O)cc1 c1(C(=O)NC2C(NCCNC(CSC)=O)C2)c(C)[nH]c(-c2ccccc2)c1C CCCCCCC(C)C(=O)NC(COCC)C(=O)NC[Si](C)(C)C N#Cc1ccc(C(=O)NC(c2ccccc2)C2CCC2)c2ccccc12 Cc1ccc(OC(C)C(=O)NC(C)(CNC(=O)C=Cc2ccsc2)CO)cc1 c1(C(N2CC(CNC(c3nc(Br)c[nH]3)=O)OCC2)=O)cn2ccnc2s1 C1(NC(CC2(C)CCCCC2)=O)CC2CC(C1)N(c1cc(C(F)(F)F)ncn1)C2 C1(CNC(CC(CC)C2CC2)=O)CC2(CC2)CN1C(C1CC2(CCO1)CC2)=O N1(C(C(C(CC)O)C)=O)CCN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(Cc2ccc(C)s2)=O)CCOC2CN(C(=O)C(O)CCC(C)C)CC12 CCC(C)C(O)C(=O)N1CCC(CNC(=O)C(CCO)N(C)C)C12CC2 C12(C(=O)NC3CCC(NC(CC(C)n4ccnc4)=O)CC3)C(=O)C3CCC1C2C3 C#CC1(C(=O)NCC2=NOC(C)C2)CCN(C(=O)C(COC)N(C)C)C1 N1(C(c2cccc(OCC)c2)=O)CCC(CNC(=O)COc2ccon2)CC1C c1(C(=O)NC(CC(C)NC(C(CCOC)C)=O)C)ccc(F)c(Cl)c1 CC(C)C(C(=O)NC(C)(CSC)C1CN(C(=O)C(O)C2CCC2)C1)NC=O.C1CC1 Cc1c(NC2CCOCC2)ncnc1N1CCC(C)C(CO)C1 N1(C(c2sc(C)c(O)n2)=O)CC(NC(c2ccccc2CO)=O)CCC1C c1(C(C)=O)ccc2nc(CNC(C(C)C)C3CCCC3)sc2c1 c1(CN(C(C(C)(C)n2cnnc2)=O)CCC(=O)N2CC(OC)C2)cccc(CO)c1 c1(C(=O)NCCN(C(c2cc(C)c(Cl)cc2F)=O)C)cccc([N+](=O)[O-])c1Cl N1(C(c2cnc3n[nH]c(C)c3c2)=O)CCOC2(CCN(C(=O)C(C)(O)CO)C2)C1 C1(F)(CNC(C2CC2(Cl)Cl)=O)CN(C(=O)C(CN2CCCC2)c2ccccc2)C1 n1(CC(C)O)cc(C(=O)NCCCCCNC(c2ccc[n+]([O-])c2)=O)ccc1=O S(=O)(=O)(CCC(=O)N1CCC(C)(n2cc(C3CCC(F)(F)CC3)nn2)C1)NCC C1(CC(=O)NC2(C(C)=O)CC2)CC(NC(c2cnc(S)nc2)=O)C1(C)C N#Cc1ccc2c(c1)CCC(NC(C1CCC(N)C1)=O)C2 CCCC(=O)N(CC(C)NC(CC(F)(F)F)=O)C Cc1cnc(C(F)(F)F)c(C(N2CCN(C(=O)CC(C)F)C(C3CCC3)C2)=O)c1 C1(NC(C(CN(C)C)O)=O)COC2(C1)CN(C(c1csc(=N)[nH]1)=O)C2 C1(C(=O)N(C2(C3N(C(C(C)(C)C)=O)CCC3)CC2)CCC2CC2)CCCN(S(N)(=O)=O)C1.C1(C)CC1 CCCCCCCCn1cc(C2CCCCN2C(=O)Nc2nn(C)cc2N)nn1 N1(C(C2(C(C)(F)F)CC2)=O)CC2CC(C1)N(C(=O)CC(N1CCCCCC1)=O)C2 CN=c1nc(C(N2CCC(NC(=O)CC3CCC(=O)NC3)C(F)C2)=O)cc(C)[nH]1 N1(C(CCCOCC=C)=O)CCc2sccc2C1CNC(C1CC1C(=O)NC)=O CC(C)CC(O)C(C)C(=O)NC(C)(C)C(C)CC(=O)N(C(C)CS(C)=O)C N1(C(CCNC(C)=O)=O)CCC(C(C(C)C)NC(=O)Cc2cc[nH]n2)CC1 CCC(C)(C)C(C)CC(=O)NC(C)C(CO)NC(c1cc(=O)c(OC)c[nH]1)=O c1(C(N2C3CN(Cc4cccc(Cl)c4)CC23)=O)ccc2c(c1)CCO2 Cc1ccncc1CNC(C1CCCCN1C(c1cc(C2CC2)no1)=O)=O Cc1cccc2c(=O)c(C(=O)NC3CCN(C(=O)C(N)=O)CC3F)c[nH]c12 C1(CCC(=O)NCc2cc(OC)ns2)CCCCN(C(=O)C=CCO)C1 c1(C(=O)NCC23C(CN(C(CSCC=C)=O)C2)C3)c(N)cc(Cl)cc1Cl N(C1CCc2c(O)cccc21)C(=O)NCC(c1cc(F)ccc1Br)F c1(C(=O)NCc2ccc(CCNC(C(CCC)C)=O)cc2)scc2c1OCCO2 c1(SC)cc(C(=O)NC2CCCC2NC(c2ccc(N)c(N)n2)=O)cc(Cl)c1 N1(C(C2C(C)(C)C2(C)C)=O)CC(NC(=O)CCCOc2cccnc2)CC(O)C1 C1(C(=O)NC(C)CCCN=[N+]=[N-])(COC)C=CCN1C(=O)C=CC(F)F C(=O)(CCC(=O)NCCCCNC(C1CCCN(C(=O)CCC)C1)=O)NC N1(C(C2(OCC)CC2)=O)CCOC(C(=O)NC2CC(=O)N(C)C2=O)CC1 C1(C(N2CC3CCC2CN3C(C2CCC3CC23)=O)=O)COc2cc(F)ccc2C1 c1(CCC=C)ccc(-c2ccc(C(N3CCOCC3C)C(=O)NCC)cc2)cc1 c1(C(N(CCCNC(=O)C2=CCC2)C)=O)ccc(O)nc1Cl c1(C(=O)NC2CCCC2C(=O)Nc2cccc(CC3CCC3)c2)cc(Cl)ncc1F C(=O)(C(F)CC(C)(C)C)NCC1(O)CCN(C(C2CCC(C(=O)OC)O2)=O)C1 c1(C(=O)NC2CCC(N(C(=O)Cc3ccoc3)C)C2)cncc(C(N)=O)c1 C1(OC)CC2(CCC(C(=O)NCC=CCNC(C3(C)CNC(=O)C3)=O)CC2)C1 N1(C(CN(CC)CC)=O)CCC(C)C1CNC(=O)COc1cccc(Cl)c1 C1(NC(C(CC=CC)C)=O)CC=C(C(=O)NC(c2ncnn2CC)C)C1 C=CCCCCCCC(=O)N1CCCC(C(=O)NC2CON(CC)C2=O)C1C c1(C(N2CCCC(CNC(C(C)N(CC)CC)=O)(CO)C2)=O)ccc(C)c(F)c1F Cc1sc2ccccc2c1C(=O)N(C1CN(C(=O)C(C)CC(F)F)CC1O)C c1(COCCC(C)NC2CCS(=O)CC2)cnc(-c2cccs2)nc1O N1(C(C2C(C)(Br)C2)=O)CC2CCC1C1CN(c3nc(-c4ccccc4)ns3)CC21 N1(C(C2CC(O)(CC#C)C2)=O)CCCCC(C(=O)NCCCC(O)CO)C1 n1(CC)cc(CC(=O)NC(C(=O)N(C)Cc2cc(C)on2)C2CCOC2)c(C)n1 C1(CC)CC(CC(=O)NCC(CC(C)C)NC(=O)CCc2cnn(C)c2)CCO1 Cc1cc(N2CCC(C(F)C(N)=O)CC2)nc(NC(c2cn(C)cn2)C)n1 Cc1nccn1CCC(=O)NCCOCCC(=O)NCC1CCC1C c1(C(=O)NCC2(CNC(=O)Cn3ncccc3=O)CC2)cc(F)c(F)cc1Cl Cc1nc(C(N2CCC(O)C2C(N2CCC(c3cnco3)C2)=O)=O)c(C)s1 C(=O)(CCCC(F)F)N(CC(CC)NC(C1CC(C(C)C)C1)=O)C C1(C)(CNC(=O)NC2CC(C)(C)OCC2)CCS(=O)(=O)N1C C1(CNC(C(=Cc2ccco2)C)=O)CCCCC1NC(C1CC(=O)N1)=O C1(CCC(=O)NCC(C)CN(C(=O)CCC2CCC(=O)NC2)C)NC(=O)NC1=O C(=O)(C(CNC(=O)CN1CCC(=O)CC1)C(C)(C)C)NC(C(=O)OC)(C)C1CC1 N1(C(C2(CC)CCCC2O)=O)CCCN(C(=O)Cc2ccc(OC)nc2)CC1 N12CC(CCC1C)C(=O)NCC(=O)N1CC3CC3C1C2=O.CCC=O.OC C1(NC(c2ncn(CC)c2)=O)CC=CCC1C(=O)NCC1(O)CCCOC1 C(=O)(C(C)C(C)S(C)(=O)=O)Nc1oc(C(=O)NCC23CC(NC(C)=O)(C2)C3)nc1C CC(CC(=O)NCC12CCC(NC(=O)C(F)=C3CCCC3)(CC1)CO2)C(C)(C)C N1(c2cc(N(C)Cc3ccc(F)c(C)c3)nc(C)n2)CC(C)S(=O)CC(C)C1 CC1COCCN(C(C2CC(F)(F)CN2C(C2CCN(C)C2)=O)=O)C1 C12(CNC(C(C3(C)CC3)NC(C(CCC)F)=O)=O)CCN(CC1)CC2 c1(C(C)C)n[nH]c(=NC(CNC(=O)C(C)c2ccsc2)C(C)C(C)C)o1 C(=O)(C1=Cc2ccccc2C1)N(C)CC1CCN(C(c2c(CC)nc(C)o2)=O)C1 O=S(=O)(CCCNc1ccc(SC2CCOC2Cl)cc1)c1ccccc1 N1(C(C2(C)N(C(c3nccc(C)c3)=O)CC2)=O)CC2(C1)CN(C)C2 c1(C(=O)NC2CC(OC)CN(C(=O)C(F)C(C)C)C2)c(C)cc(C)oc1=O CCC(O)CCN=c1nc(N2CCCC(C(=O)NC(C)(C)C)C2)c2sccc2[nH]1 N1(C(CN(C(C)C)C)=O)CC(O)CC1C(N)=O.C12CC(O)C1CC(=O)N2 C1(NC(CCc2onc(C)n2)=O)CN(C(C2CC(F)(CO)C2)=O)CC1C C1(CC=C)(NC(=O)C2CC2)CCN(C(=O)C(C2CC2)OC)CC1 NS(=O)(=O)CCC(=O)NCC1(CNC(C2CCCCC2F)=O)CC12CCC2 C12(COC)CC(NC(=O)CC(=O)N(C)C)(CN1C(c1cnc(O)c(OC)c1)=O)C2 C1(=CCNC(C2(CCOC)CC2)=O)CCN(C(=O)C(=O)N(C)C)CC1 C1(CNC(C(C(C)C)(C)O)=O)CCC2(CN(C(=O)CCn3cnnn3)C2)O1 c1(C(=O)NCC2(CNC(C3CCC(CC)C3)=O)CC2)sc([N+](=O)[O-])cc1Cl CC(C)C(C(=O)N1CC(CCNC(C2CCO2)=O)C1)N1CCCCC1 C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCN(C(C2CCC=CCC2)=O)CC1O N1(C(c2c(CC)n[nH]c2)=O)CCCCC1C(=O)NCCCC(=O)NC(C)C c1(C(N2CCC(C(C)(C)NC(=O)C3=C(Cl)CC3)C2)=O)cc2c(cc1Cl)OCO2 C1(NC(c2c(C(=O)OC)cco2)=O)CC2CC(NC(=O)CCOC3CCC3)C1C2 Cc1cc(C)c(C=CC(=O)NCC2CC2NC(=O)CCC2CC2)c(C)c1 C(C1=CCN(C(c2ccn(C)c2C2CCC2)=O)CC1)NC(CCSCCCC)=O C1(OC(C(c2cccc(O)n2)C)=O)CCN(c2ccc(Cl)cc2)C1=O c1(NC(C(C)=C2CCC2)=O)ccnc(Oc2cccs2)c1.C12CCC1CNC2=O C1(NC(C2C(C(=O)NCC3(C(=O)OCC)COC3)C2)=O)CNC(=O)N1 CC1(C)CC(NC(=O)CCC2CC2(C)C)CN(c2cnc(C#N)cn2)C1 CC(N=c1[nH]c2c(c(=NC3CC(C4CC4)C3)[nH]1)CCCCCC2)c1nc(=N)[nH][nH]1 C1(NC(=O)C=CC(C)C)CCCC(C(=O)NC2(Cc3cscc3Br)CCC2)C1 CC1(C)CCC(C(=O)NCCCOCCNC(C2CNC(=O)N2)=O)OC1 Cc1cc(C)c2c(c1)CN(C(=O)CCCC1CCCCC1=O)CC2 C1(NC(CNC(C)=O)=O)C2CC3CN(C(=O)Nc4ccccc4O)C1C3C2 c12ccc(c(OC)c1)CN(CC)C2C(=O)NC(C)(C)CC.N1(CC)CCCCC1 Cn1cnc(N2CCC(OCCCNC(c3nc(Cl)ccc3F)=O)CC2)cc1=O C(=O)(CS(=O)(=O)C1CC1)N(CCn1cc(Cc2ccc(Br)cn2)nn1)CC N1(C(C(C)OCC)=O)CCC(OC)C1.c1(N2C(C)COCC2=O)nn[nH]n1 CC(C)C(CNC(=O)C=Cc1cnn(C)c1)C(=O)N(C1(C)CCCC1)C C(c1scnc1C)=CC(=O)NC1C(NC(C(C)(c2cccs2)N(C)C)=O)COC1 N1(C(c2c(C)ncc(N)c2)=O)CCC(C)N(C(c2coc(S(C)(=O)=O)c2)=O)CC1 N1(C(CC(C)(C)C)=O)CCN(C(=O)COc2ccccc2O)CC1CS(C)(=O)=O C1(C(=O)NCC(C)OCC=C)(CNC(c2nnsc2N)=O)CCCCC1 c1(OCC(=O)NCC2CN(C(=O)Cc3c[nH]nc3O)C2)ccccn1 c1(C(N2CC(NC(Cc3cnc(C)[nH]3)=O)(CO)C2)=O)cnncc1C N1(C(C2(NC(CC(C)OC)=O)CCN(C)C2)=O)CCn2nc(C)cc2C1 Cc1nc(C(=O)NC2CC(CC(=O)NCC(C3CC3)C3CC3)C2)c(C)s1 N1(C(c2cc(Cl)cs2)=O)CCC2(CC1)CC(C(N1CCC1CO)=O)CO2 c1(NC(C2C3CN(Cc4cn(CCC)nc4)C2C3)=O)cc(O)cc(O)c1 c1(C(=O)NCC2CCN(C3CC3)C2)c(O)nnc2c1CCC2 CCC(CC(C)C)C(=O)N1CC2CC1(C(=O)NCC1(CCCO)CC1)C2 c1(NC(C2CCNCC2CO)=O)ccc(OC(F)(F)F)cc1 C1(C(N2C(CCNC(=O)CCF)CSCC2)=O)CC2CCCC(C1)C2=O CC1CCN(C(c2[nH]nnc2C2CC2)=O)CC1CNC(c1cc[nH]c(=N)c1)=O c1(CC)cc(C)c(C(=O)NC2(C(=O)NC3CC3(C)C(F)F)CCC2)o1 c1(C(N(CC(C)CNC(C2(F)CCS(=O)(=O)C2)=O)C)=O)sc2nccnc2c1N Cc1nc2ccccn2c1C(=O)NCC1CCCN1C(c1ncn2c1CCC2)=O C1(CC(N2CCOC(CNC(C3(C4CCCO4)CC3)=O)C2)=O)NC(=O)NC1=O C#CC1(NC(c2ccc(CNC(=O)C(CCC)N(C)C)s2)=O)CCCCCC1 C=CCCCCCCC(=O)NC(C)CCCNC(=O)C(n1ccc(C2CC2)n1)C S(=O)(=O)(c1ccc([N+](=O)[O-])cc1C(=O)O)N1C2CCN(CCOC)CC2CCC1 C1(NC(NC(CC)CSC)=S)CCCC(C)C1C C1(N=c2cc(Br)n(C)[nH]2)(c2n(CCOC)nnn2)CC2(CC2)C12CCC2 CC(C)C(CNC(C1CCN(C)CC1)=O)C(=O)NCC1CCCCO1 N1(C(C=NS(N(C)C)(=O)=O)=O)CC=CC(NC(C2CC2(C)Br)=O)C1 C(C(O)CC(=O)N1CCC(OCCN(C)C)C1)NC(C=C(C)C(F)F)=O C(=O)(CS(=O)(=O)CC)NC(CCN(C(CC(CC)C)=O)C)c1cccs1 Cc1ccc(C(N2CCCN(c3ncc4c(n3)CCOC4)CC2)=O)cc1[N+](=O)[O-] N1(C(COC2(C)CN(C(c3c(OC)nsc3)=O)C2)=O)CC(CO)OC(C)C1 c1(CC(=O)NCCC(C)NC(c2ccc(C)cc2Cl)=O)csc2cc(C)sc12 n1(CC(N2CC(C)N(C(c3cccnc3)=O)CC2)=O)cc([N+](=O)[O-])c(O)nc1=O C(=O)(C(C)(C)C(C)(F)F)N1CC(CC(C(=O)NCC(C)(C)F)F)C1 c1(-n2c(C(C)(CCCl)n3cc(CN4CCCC4)nn3)nnn2)ccccc1Br c1(C(N(CC(CN(C(C(C(C)(C)C)OC)=O)C)O)C)=O)c(F)ccc(C)c1Cl c1(C2(Cc3cc(C(=O)NC4CC5CCC4N5)ncn3)CC2)ncc(Cl)cc1F N1(C(c2cccc(OC)c2)=O)CCCC2C1CCN2Cc1ccc(CSC)cc1 N1(C(c2cn(CC)nc2)=O)CCN(C(=O)C=C2CCN(C)C2)CC1CF c1(C(N(C2CCS(=O)(=O)C2)CC=C)=O)cc(S(=O)(=O)CC)ccc1OC N1(C(C(CNC(c2c(CC)nccc2)=O)O)=O)CCC2CCCC12 C(=O)(CC1CNc2ccccc21)N(C)CC1CN(C(=O)C=Cc2cccnc2)C1 N1(C(C2CCCCS2(=O)=O)=O)CCn2cccc2C1c1ccc(Cl)cc1 N1(C(CC=CC=C)=O)CC2CCC1C1CN(C(c3c(C)noc3N)=O)CC21 C1(NC(c2nnc(O)nc2O)=O)CN(C(=O)CCCn2ccnn2)CCC1CO C1(NC(c2cccnc2C)c2n(CCCSCC)nnn2)CCCN2CCCC12 Cc1ccc(CC(=O)NC2CCC(CCNC(C3(CC(F)F)CCC3)=O)C2)o1 C1(C(N(CC(C)NC(CCC)=O)C)=O)N(C(=O)OC(C)(C)C)CCC12CC2 S(=O)(=O)(c1cccc(Br)c1F)N1C(C(C(N2C3CCC2CC3)=O)C2CC2)CCC1 N1(C(C)C2CC2)CC(C(N2CCC(O)(CNC(c3cnn(C)c3)=O)C2)=O)CC1=O C1(NC(=O)CCOCc2ccccc2)COC2CN(C(=O)CCC3CC3)CC12 C12(NC(C(CC)CC)=O)CCC(CN(C(C3CCCS(=O)(=O)N3)=O)C1)C2 N12CC=CC1C2=O.C12CCC1C(=O)NC2.N1(OC)CCC1CC1CC1 N1(C(C(n2ncc(C)c2)C)=O)CC(O)CCC1C(=O)NC1CCCCC1 N1(C(C)=O)CCCC(NC(c2coc(CNC(C3(C(C)(F)F)CC3)=O)n2)=O)C1 CCC(CC)(CCC(=O)OC)NC(c1c(C)cc(Cl)cc1C)=O C(CN=c1nc(CN2CCCCC2CCO)[nH]s1)=NC(C1CCC(CC)CC1)=O N1(C(CCC#C)=O)CC(C2CCCN(C(C3CCCCN3N=O)=O)C2)C1 Cc1occc1CNC(C12CC(NC(c3ccn(C4CC4)n3)=O)(C1)C2)=O CN1CCCC1(C)C(=O)NNC(=O)C1CCNC1c1ccccc1 N1(C(C)C)CCN(CCCC(N2CCC(NC(=O)CC(C)O)C2C)=O)CC1 Cc1csc(CC(=O)NCC(C2CCCC2)NC(=O)Cc2csc(C)n2)c1 C1(C(=O)NCCC2(CNC(C3(OC)CCOC3)=O)CC2)COCCN1CC(F)F N1(C(c2c(Br)cn(CC)n2)=O)CCC(CNC(C2CCOC2)=O)C(O)C1 C12CCCCC1NC2=O.c1(C(=O)NCC(CN(C)C)(C)C)ccc(C(F)F)cc1 C(=O)(CCCC(C)(C)NC(c1ccccc1OC)=O)NCC#C c1(OC)cc(C(=O)NC(CNC(C2(O)CCCCC2)=O)CC(F)(F)F)cc(F)n1 N1(C(C(C)(C)O)=O)CCC2(CCCN(C(c3cc(Cl)nc(Cl)c3)=O)C2)C1 c1(SCCC)cccc(C(=O)NC2CCC(CNC(=O)Cn3cncc3C)C2)c1 C1(C(=O)NCC(c2cccs2)C)CCN(C(C2CC2C(C)(F)F)=O)CCO1 C(=O)(C(CC)(CC)CC)NC1CCCN(C(c2nc(CC)oc2C)=O)C1 N1(C(c2c(C)coc2)=O)CCC2(CC2C(=O)NCc2cccnc2C)C1 c1(CNCCc2scc(C)n2)c(C)nsc1C.c12cc(on1)S2 Cc1ccc(CCC(=O)NC2CCC2NC(C2CN(C)C(=O)N2)=O)cc1C CCC(C(=O)N1CC(N2CCCC2=O)C1)C(C)(C)CC.c12cn(C)nc1C(=O)NC2 c1(C(=O)NCCN(C(c2c(C)cn(C)n2)=O)C)nc2ncccn2n1 C(C(C)(C(=O)OC(C)(C)C)NCC(c1ccccc1)N(C)C(C)=O)SC Cc1nnccc1C(=O)NCC1(NC(=O)COC2CCOC2)CCCC1 CCCCC(O)C(C)C(=O)N1CCC(C2CC2)C1C(=O)NCCCN1CCCC1 CC1C(NC(C2CCN2C)=O)CC2CCC1N2C(=O)COC1CCOCC1 c1(CC(N2CCC(CC(=O)N(CCCCC=C)C)C2)=O)c(C)noc1C N1(C(C2C(C(C)(C)C)C2)=O)CC2(C(N3CC(O)C(N=[N+]=[N-])C3)=O)CCC1CC2 n1(CC(=O)NC2C(NC(c3ocnc3C3CC3)=O)CC2)cnoc1=O C1(OCC#C)CCN(C(c2cnn(CC)n2)C(=O)NCCCC2CC2)CC1 c1(NC(C2CCN(C(Cn3nnc(C)n3)=O)C2)=O)cc2ccccn2c1 C(=O)(CC(O)(C(F)(F)F)c1ccccc1)Nc1ccc(-n2c(C)cnn2)cc1 c1(C(N2CC3C(C(=O)Nc4cc(C(=O)NC)ncc4)C3C2)=O)cccc(=O)n1C c1(C(N2CCC(N(C(=O)CSc3n[nH]c(O)n3)C)C2)=O)cccc([N+](=O)[O-])c1Cl C(=O)(C(C(C)NC(c1coc(CO)c1)=O)C(C)C)NC(CC(=O)OCC)C N1(C(C2C(C)CCO2)=O)CCN(c2ccc(C(=O)N(CCO)CCO)cn2)CC1 c1(C(=O)NC(CC)C(=O)OC)ccc2c(-c3cccc(OCCF)c3)n[nH]c2c1 c1(C(N(C2CCN(c3nc(O)c(C)s3)C2)CCC)=O)cc(O)nc(C)n1 C=CCCCC(C1CC1)NC(C1CCN(C(C2OCCC2C)=O)CC1)=O C(N=c1nc2scnc2c(NC2CCSC(C)(C)C2)[nH]1)c1c(=O)ccn(C)c1 c1(C(=O)NCC(CO)NC(C2CN(c3nncs3)C2)=O)cc(F)c(O)c(F)c1 C=CC1(C(N2CC(OC3(CSC)CC3)C2)=O)CCCCC1.C12CCN(CC1)C2=O N1(C(CCCN(C(C)=O)C)=O)CC2CC1CN2Cc1ncnn1C(C)(C)C N1(C(C(c2ccc(C)cc2)=O)=O)C2CCC1CC(NC(c1coc(Br)c1)=O)C2 C1(C(N2C(C(=O)NCc3occ(C)n3)CC(C)C2)=O)CN(C)CC(C)O1 c1(NC(CC2CCCN(Cc3ccc(OC)nc3)C2)=O)cccc(C#N)c1C C1(CNC(=O)C(C2CCCCC2)F)(NC(C2CC2C2CCCO2)=O)CCOCC1 c1(CC(=O)N(CCNC(c2ccc(C)cc2)=O)CC)cc[nH]c(=N)c1 N1(C(CN2CC(C)(C)C2)=O)CC(O)CC1(C)C(=O)NCc1ccccn1 Cc1nc(C(=O)N(CCNC(=O)C(C)CC(C)C)C(C)C)ccc1C#N C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)C=CCN(C(=O)Cc2cn[nH]c2)C1 O(N1CCC(CC(=O)NC(C)C(C)NC(=O)Cc2noc(C)c2C#N)CC1)CC c1(OC)ccc(F)c(N)c1C(=O)NC1CC(CNC(=O)C=Cc2ccccc2)C1 CC1CN(C(C2CCC(O)CC2)=O)CCCN1C(c1cnnc(Cl)c1)=O c1(C(=O)NCC(CNC(C(CC=CCC)C)=O)(C)F)cc(N)c(O)c(F)c1 C(=O)(C(CCN(C)C)NC(c1ccncc1F)=O)N(C)CCO.C1(N(C)C)(C(=O)O)CC1 c1(C(=O)NC23CC(NC(C(C4CCC4)OC)=O)(C2)C3)csc2cc(OC)ccc12 c1(C(=O)NCCOCCCNC(C2CC2Cl)=O)ccc(SC(F)F)cn1 CC1CCC(=CC(N2CCC(O)(CCNC(C3(Br)CC3)=O)C2)=O)CC1 C1(C(N2C(C(N(C)C)=O)CC2)=O)COCCN(C(C2CC3(CC(=O)C3)C2)=O)C1 C(C)(C(=O)N(CCNC(C1CCCO1)=O)C(CC1CC1)(C)CC)OCCC#C CCCC(C)CC(=O)N(CC(C)(C)NC(=O)C=C1CCC(c2ccccc2)C1)C C1(CNC(c2cc(C(=O)OC)on2)=O)CCCCN(C(C2(C)CCC(C)C2)=O)C1 CC1CC(NC(c2c[nH]ccc2=N)=O)CN1C(c1cc(C2CC2)oc1C1CC1)=O CC1CCC(C(=O)NCCc2csnn2)CN1C(=O)CCOCC(F)F C(CC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1cc(Br)sn1)=O)OC C1(CC(=O)NC2CC(CNC(c3cc(CCC)[nH]n3)=O)C2)(CC#N)CNC(=O)C1 c1(OCC(C)NC(=O)Nc2ccsc2CC2CC2)c(F)cccc1F C1(C(=O)Nc2cccc(NC(C3C(c4n(C)nnc4)C3)=O)c2)CCOCC1(C)C c1(C2(C)CC2)nc(Cl)cc(=NCC2(CNC(=O)CCCC3CCC3)COC2)[nH]1 C1(C(=O)OC)C(C)CCN1C(c1ccc(CN=[N+]=[N-])cc1)=O c1(C(=O)NCCC2CC(NC(C3(CC)CCC3)=O)C2)oc(CO)cc1C C(=O)(C1CCc2c[nH]nc21)N1CCCC(CC)CC1.C1(=O)CON1CC c1(C(=O)NC(C2(O)CCN(C(C(C)NC(=O)NC)=O)C2)C)ccn2ccnc2c1 C(=O)(C(CC#CC)NC(=O)C=Cc1cc[nH]c1)NC(CCC=C)(C)C Cc1nc(N2CCCC2c2ccc(-c3ccccc3)cc2)sc1Br Cc1c(CC(N2CCCC(CNC(c3cc(Cl)no3)=O)C2)=O)sc2ccccc12 CCC(C)C(O)CC(=O)NCc1ccsc1C(=O)NC1CCS(=O)CC1 N1(C(C2(C)CC(=O)C2)=O)CCN(C(C2(C#N)CC3CC3C2)=O)CC(O)C1 S(=O)(=O)(c1cccc([N+](=O)[O-])c1C)Nc1c(NC(=O)OC(C)(C)C)ccnc1F c1(OC)cc(C(=O)NC(C)(CNC(C2(O)CC2(C)C)=O)CO)cc(OC)c1C N1(C(C2N(CC)C(=O)CCC2)=O)CCC2CN(C(C34CC(CN3C3CC3)C4)=O)C2C1 C=CC(CC)C(=O)NCC1CCN(C(=O)CN(C)C(=O)C2CC2)C1 C1(NC(C2(N3CCN(C)CC3)CC2)=O)CN(C(=O)CC2CCC2)CC2(CC2)C1 N1(C(C(CCC)N(C)C)=O)CC2CC(C1)N(C(c1csc(C3CC3)n1)=O)C2 CC1(O)CCC(CC(=O)NC2C3CC2N(C(C2CCCO2)=O)C3)CC1 C(=O)(CC(F)(F)C(F)(F)F)NCC(C12CCC(CC1)C2)NC(=O)C(F)=CC1CC1 N1(C(CCC(C)SC)=O)CCCCCC1C(=O)NCC1(C)CCC(=O)N1 C1(C(N(CC(C)NC(COc2c(C)occc2=O)=O)C)=O)CCc2ncnn2C1 CC(C)CCCC(=O)NC1CC2C(C(=O)NCC3CCCCCN3C)C2C1 S(=O)(=O)(C1CC2(CC2)C1)N1CCCC(C(N2CCCC(C(N)=O)C2)=O)C1 N1(C(CCCC=C)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(C)C1C CCC(CC)CCCC(=O)NCC1CC1C(=O)NCC.C12CCCCN1C2 C(CC)(CCC(=O)OC)NC(C(CC=C)N1CCC(C)CC1)=O c1(CC)ccc(C(=O)NCC2CCN(C(=O)Cc3ccc(C)o3)C2)cc1F c1(C2CCN(c3cc(NC(CC=C)CC=C)ncn3)CC2)cccc(C#N)c1 c1(C(N2CC(CC(C)NC(C(C(CC)C)OC)=O)C2)=O)cc2cccnc2[nH]1 c1(C(N(CC(CC)OC)C)=O)coc(CNC(=O)C(COC)N(C)C)n1 Cc1cc(C(=O)NC2CCC(NC(C3CCC3)=O)CC2)oc1C C1(C(=O)NC(C=C)(C)C)CCC(C)N1C(=O)C(C1CCC1)OC Cc1nn(-c2ccccc2)cc1C(=O)N(CC(O)C(C)(C)C)C C1(NC(=O)CC2CN(C(=O)C=CCN3CCC3)CCO2)CC2CC3C(C2)C13 CCC(C(=O)NOCC(=O)NC1CN(CC)CC1C)N(C)C C1(NC(c2nccc(OC)c2)=O)CN(C(=O)C(C)NC=O)CC12CC2 N1(C(c2c(OC)csc2)=O)CC(CNC(=O)CC(C)CF)C2(CCOCC2)C1 N1(C(CC(C)SC)=O)CCN(CCCCCNC(=O)Cc2cc[nH]c(=N)c2)CC1 N1(C(CC(C)F)=O)C2CC1CN(C(c1ncc[nH]1)=O)C2 c1(NC(=O)CN2CC(CO)CC(CO)C2)cc(F)c(F)cc1Cl C(C(=O)NCC(C1CCN(C(C2(C)CC2)=O)CC1)(C)O)(C(C)C)OC CC1(C)CC(CNC(c2ccccc2Cl)c2nnnn2CCC2CC2)CNC1=O C12(CNC(C=C(C)C3CC3)=O)CCC(CC1NC(=O)Cc1cc(F)ccc1F)C2 CCC(C)C(=O)C(=O)NCCC1(O)CCN(C(c2cc(C)sn2)=O)CC1 C1(C2CC2)(CNC(c2n(C=C)ncc2)=O)CCN(C(c2cc(C)ncc2C)=O)C1 N1(C(c2coc(CO)c2)=O)CCC(c2ccc(Br)cc2)NC1=O c1(C(=O)NC(C2(O)CN(C(C3CC(OC)C3)=O)C2)C)sc(Cl)cc1Cl C1(NC(C2CC2C(F)(F)F)=O)CCN(C(=O)CCc2csnn2)C12CCC2 N1(C(CC2C=CC(NC(c3c(C)cccn3)=O)C2)=O)CCC(C)(C2CC2)C1 Cc1ccc(CC(=O)NC(C)(C(N2CCCC2CCC(C)C)=O)C2CCC2)o1 CCC(CC(=O)NC(c1ccsc1)C)NC(=O)Cc1csnc1C C1(NC(C(N2CC(CC)SCC2)=O)=O)CCOC12CCOCC2 N1(C(CN(C)C(N)=O)=O)CCC(C2CCN(C(c3cc(C4CC4)ccn3)=O)C2)C1 c1(C(=O)NC(c2cccnc2)C(=O)NCCC(C)OC)c[nH]ccc1=O C12(NC(=O)CCF)CCCN(CC(F)(F)F)CC1C2.c12cccc(c1)NC2=O c1(C(=O)NC2CN(C(CCc3ccn(C)n3)=O)CC3C2C3)csc2c1CCCC2 c1(N2CCC([SH](C)C3CC3)C2)nc(-c2ccccc2)nc(=NCCC=CBr)[nH]1 N1(C(C)=O)CCCC12CCN(C(=O)CC)C2.C(C(C)C)N(C(C)CO)CCC1CC1 C1(C(N(C2COCC2(C)C)CC)=O)CCN(C(=O)CC2(C)CCOC2)C(C)(C)C1 N1(C(C2ON=C(C)C2)=O)CCC(N(CCO)C(C2(C)CS(=O)(=O)C2)=O)CC1 N1(C(c2cnc(=N)[nH]c2)=O)CCC2CC(NC(c3cc(Cl)sc3Cl)=O)CCC2C1 c1(C(=O)NC(CNC(C(C)n2ccnc2)=O)(C)C2CC2)ccc2c(c1)nnn2C c1(C(=O)NCC(CC(C)C)NC(C2(C)CC2C)=O)cnc(N)c(Cl)c1 C(CCC(O)C(=O)N1CCCN(CCO)CC1)NC(=O)CCc1cnn[nH]1 c1(CC)cc(NC2CN(C(c3n[nH]cc3C)=O)CC2C)nc(C)n1 CCC(C)(CCNC(=O)Cc1ccc(O)nc1)NC(=O)C(=Cc1cccnc1)C c1(SC)ccc(NC(C2CC(NC(=O)CN(C)C)CCO2)=O)cc1 Cc1cc(Cl)cc(N)c1C(N1CCC(C(C)(C)C)C1)=O CC(C)C(C)CC(=O)NC1(CNC(c2ccc(Cl)cc2Cl)=O)CCOC1 c1(CNC(=O)CCc2cnc(O)[nH]2)ccc(C(=O)NCc2cccnc2)cn1 C1(F)(CNC(c2n(C(C)C)ccn2)=O)CCN(C(C2CCC(C)(F)CC2)=O)CC1 c1(C(=O)NCC(C)N(C(=O)CCNC(N)=O)CC)c(F)cncc1F c1(C(=O)NC(C(C)NC(=O)Cc2cn[nH]c2)(C)C)cccc(S(N)(=O)=O)c1 N1(C(c2c(C)nc(O)cc2)=O)CCC(C)(C)C(C(N2CCN(C)C(CO)C2)=O)C1 Cc1occc1C(N1CCCC1CCNC(C1CC1(C)C(F)F)=O)=O S(=O)(=O)(c1ncc[nH]1)NC1CC(C(=O)OC)C(c2nncn2C)C1 C1(NC(C2CCCN(C(CC3CCCC(C)(C)C3)=O)C2)=O)CN2CCC1(C)CC2 S(=O)(=O)(c1ccc(C(=O)N(C)C(C)C)cc1)NCCCC.c12cccc(c1)NC2 C(=O)(C#CC1CCCCC1)NCC1CCCCN(C(CCC2N(C)CCC2)=O)C1 c1(C(N(CCNC(C2CCC(OC)C2)=O)C(C)C)=O)cc2cccc(Cl)c2cn1 Cc1ccnc(C(=O)N(C)CC2CN(C(=O)C(n3ccnc3C)C)CCO2)n1 c1(C(=O)OCC)cc(C)ccc1S(=O)(=O)Oc1cccc(OC(C)C(C)C)c1 N1(C(c2cccc(C)c2)=O)CC2(CCCC2NC(C2CC3CCC2C3)=O)C1 C=CC1(C(=O)NC2C(O)C3CCOC23)CCN(C(C2CC(OC)C2)=O)C1 N1(C(c2c(C(=O)OC)ccs2)=O)CC2(NC(c3cc(C4CC4)ccn3)=O)CC1C2 N1(C(C(CCC)C)=O)CCC(CNC(c2cc(C)cc(F)c2)=O)C(F)(F)CC1 c1(N(C2CCCNCC2)C(c2cc(C(F)(F)F)c[nH]2)=O)ncnc2sc(Br)cc12 C1(NC(CNC(=O)OC)=O)CC2CC1CC2C(=O)NCC(F)C1CCC1 N1(C(c2cc(OC)n[nH]2)=O)CC2C(C1C(N1CCCC1C(N)=O)=O)C2(C)C CC1CN(C(C2(C#N)CC2)=O)CC1NC(=O)COc1ccccc1 c1(CCC)cc(=NC2C3CCC2(C)C2(OC)CC3C2)[nH]c(Cl)n1 c1(C(=O)NC2CCCC(NC(c3cc(C(C)C)on3)=O)C2)cnc(Cl)cc1N S(=O)(=O)(c1cc(CC)c(F)cc1OC)N1CCCN(CC)CC1C Cc1cc(O)c(C(N2CCCC(N(C)C(C3CC(O)CN3C(N)=O)=O)C2)=O)nn1 c1(CC(=O)NC(C)C(C)NC(=O)C(Cc2ccco2)N(C)C)cccc(CO)c1 c1(NC(C23CN(C(C(C)CC(N)=O)=O)C(C2)CO3)=O)cccc2occc12 C(=O)(CCCC(C)(F)F)NC(C(C)C)CCN(C)C(c1ccsc1C(F)F)=O CCCC(O)C(=O)NCCCOCCN(C)C(C1COC(=O)N1)=O Cc1cc(C(=O)NCC2(CC(=O)NOCCCN(C)C)CCCCC2)c(C)cn1 CCCCCC(CC)C(=O)NCC1(C)CCCN(C(=O)CCOCC)C1 c1(C(=O)NCC(CC=C)NC(=O)CC(C)(C)C2CC2)ccccc1-c1nc[nH]n1 c1(N(C)C)ncnc2cc(C(=O)NCCCN(C(=O)C(N)=O)C3CC3)ccc12 N1(C(CCC2(C)CN(C(C(C(C)C)O)=O)C2)=O)CCCC(C)(C#N)C1 Cc1cnn(C)c1C(=O)NCCOC1CN(C(c2cn(C)nc2C(F)(F)F)=O)C1 C1(CNC(c2ccc(SC)o2)=O)CN(C(=O)CC(Cl)Cl)CCC1O c1(C(=O)NC23CC(C(=O)NCCc4cc(C)no4)(C2)C3)c[nH]c2ncccc12 C(C(C(C)(C)C)NC(C1(C2CCCO2)CCC1)=O)NC(c1n(C)cnc1)=O c1(C(N2CCCC(C)(NC(C(C)N(C)C)=O)C2)=O)cccc2c1C1CCC2CC1 N1(C(CC(C)SC)=O)CCCCC1CNC(c1ccc(CSC)o1)=O N1(CC(C)C)CCC(C(=O)Nc2ncccc2OCC(F)F)C(C)C1 c1(CNC(CCC)=O)ccc(C(=O)NC2CCC2NC(=O)CNC=O)cc1 C1(OC)CN(C(=O)CCC2CCCOC2)CC1NC(c1ccc(CSC)o1)=O N1(C(C(CC)CC(F)F)=O)Cc2ccnn2CC(NC(=O)C=C2CCOCC2)C1 Cc1nc(CNCC2CCC(C(=O)Nc3cnn(CC4CC4)c3)CC2)ccc1Br CCCCC(C)CCC(=O)NC(C)C(C)(C)C(=O)N1CCCC1C c1(C(N2CC(C)C(NC(=O)CC3CC=CCC3)C2)=O)cc2scnc2[nH]1 C1(CC)CCCC1(C)C(N1CC(C(=O)NCCNC(c2cc(F)n[nH]2)=O)C1)=O N1(C(c2c(C)nco2)=O)CCN(C(=O)CNC(c2c(C)n[nH]c2C)=O)CC12CC2 C1(NC(C2CCC(=C)CC2)=O)CCCC2CN(C(C3CC3C)=O)CC12 N1(C(C(COC)C)=O)CCCCC2(C1)CN(C(=O)C(C)N=c1cc[nH]cc1)C2 CCCCC(CC)CC(=O)NC1CC(NC(=O)CN(C2CCC2)C)CC1O c1(C(=O)NC(C(C)NC(C2CN(CC)C(=O)C2)=O)C)cnc2n(c1=O)CCS2 C(=O)(CCCC(F)(F)CO)NC(=O)C(O)CC(F)F.Cn1cc(C23CC2C3)nn1 c1(C(N(C2CCN(C(=O)C(C)CF)C2)CC)=O)ccc(N(C)C)nc1 C#CCC(C)(C(=O)N(CCC(=O)N1CCOCC(C2CC2)C1)OC)SC N1(C(C(C)P(C)(C)=O)=O)CC2CCC(C1)N2C(c1ccn(C2CC2)n1)=O CN=c1nc(N2CCCCC(C)(C)C2)[nH]c(=NCc2ccc(CO)o2)[nH]1 Cc1cc([N+](=O)[O-])cc(C(N2CCN(C(=O)C(C)(C)F)CC2C(C)C)=O)n1 S(=O)(=O)(c1ccc(NC(=O)NCC2CC2)c(Cl)c1)NC1C(SC)CCC1 c1(C(N(C(C)CNC(C2(C(=O)NC3CC3)CC2)=O)C)=O)c(Cl)csc1Cl C1(C(C)Nc2cccc(C(=O)NC(C)(C)C)c2)CC(C(C)(C)C)=NO1 c1(N2CCNCC2)ncc2n1CCCC2.C(CCC(=O)NC)SC C(=O)(C=C1SCC(=O)N1C)N1CCCC(C)(CNC(c2cnc(OCC)s2)=O)C1 C1(NC(CC2CC(SC)C2)=O)C2CN(C(=O)CSc3ccccc3F)CC12 CCCCCCCCNC(=O)C(N1CC(O)CC1CNC(=O)CSCC(C)C)=O C(=O)(C1=NN(CC(C)C)C(=O)CC1)NC(CC)CN(C(=O)C1=CCSC1)C C1(C(=O)NC2CCN(CCNC(CC3(C)CC3)=O)CC2)CCCCC1C1CC1 C=CCCC(F)(F)C(=O)N(C)CCC1CCCCN1C(=O)C(C)SCCCC c1(C(=O)NC2CCN(c3nc(C)cc(C)n3)C2)oc2c(C)ccc(C)c2c1C N1(C(c2c(C)c[nH]c2)=O)CC(=O)NCC1C(=O)NCCC1CCSC1 C1(CC)CCCCC1NC(C1(CNC(=O)C=Cc2cscn2)CCCC1)=O c1(CC(=O)NCC(C)(C)CNC(=O)C(C)(C)c2cnco2)c(F)cccc1F N1(C(C2(C(C)C)CC2)=O)CCCCC(CNC(=O)C(c2ccc(Cl)c(Cl)c2)C)C1 CCCC(C)(C)C(=O)N1CCC(CN(C(=O)C(C)(O)c2ccccn2)C)CC1 C1(C(=O)NC2CC(C(=O)NCCNC(C(C)C)=O)CC2O)CC12CCOCC2 C1(NC(=O)CN(C(=O)Cc2ccc(O)cn2)CC2CC2)CCOC12CCOC2 c1(CCC)cc(C(=O)NCCOCCCNC(C2CC(C)CO2)=O)nn1C C1(F)(C(=O)OCc2ccnn2C(F)(F)F)CN(CC)CC12CNC2 NS(=O)(=O)C1(CNC(C2CC2Nc2ccoc2-c2ccccc2)=O)CC1 c1(C(=O)NC2C(NC(C(C=C)(C)CC)=O)C2)ncn2ccccc12 C1(O)(CNC(COCCOCC#C)=O)CC(C(N2CCC2CC)=O)C1 c1(OC)cc(F)c(F)cc1C(N1CCC(NC(C2OCCC2C)=O)CC1)=O c1(C(N2C(COCC#N)CCCC2)=O)cnc2c(c1)CNC2=O c1(CC(=O)NC2(CNC(CC(=O)NCC)=O)CCC2)ccc(C)nc1Cl c1(COC)c(C(=O)N(CCNC(c2ccccc2CO)=O)CCO)cnn1C N1(C(c2occ(C)c2)=O)CC2CCC(NC(c3cccc(Br)c3C)=O)(C2)C1 C(CCCC(=O)Nc1ncnn1C1CC1)OCC(=O)NCC(=O)Nc1cn[nH]c1 C(C(CCC(=O)N1CCCCC1)C(C)C)N1CCCC(CC)C1 N1(CC)C(=O)CCC1C(=O)N(C)CCNC(c1ncccc1C)=O Cc1nc(O)ccc1C(=O)NCCCCC1CCCN(C(=O)Cc2cncs2)C1 C(=O)(C1=CCCN(C(C2CC(=C3CCC3)C2)=O)C1)NCc1cc(C)cc(Cl)c1 C1(CC)CN(C(c2nccs2)=O)CCC1NC(c1ccn(CC(F)(F)F)n1)=O Cc1ccccc1N1CCC(NC(C2(N)CC3CC3C2)=O)C1=O c1(C(=O)NCC2(CN(C(C3C(C)(CC)C3)=O)C)CC2)ccc2c(c1)CC2 C1(NC(C(C)C2CCOC2)=O)CCC(CNC(C2CS(=O)(=O)C2)=O)C1 C1(C(=O)NC(CC=C)C(=O)N2CCN(C(C)=O)CC2)CCC(C)(C)OC1 CC1CCCC=C1C(=O)N1CC(O)CC1C(=O)N(CCO)CCO C=CC1CN(C(c2ccc(SC3CC3)cc2)=O)CC1NC(=O)C(F)=CCCF CCC(C)CC(C)C(=O)N(C)CC1COCCN1C(=O)Cc1cc[nH]c1 O1NC(=O)C(C(C)C)CNC(=O)C1.c1(OC)ccc(N(C)C)cc1 N1(CC(N2C(CNC(c3cccn3C)=O)CC(OC)C2)=O)C(=O)CC(C)(C)C1=O c1(CN2C(CC(=O)NC(c3cccc(OC(F)F)c3)C)CCC2)noc2c1CCC2 N1(CCC(=O)NCC(=O)N(CC#N)CC#N)CCOCC1 Cc1noc(Cl)c1CC(=O)NCCC1CN(C(=O)C(C)C(F)F)CCO1 C(C)(C(=O)N(CCCCN(C(=O)C(C1CCC1)C1CCC1)C)C)NC(CC)=O C1(CCNC(C(n2c(C)ccn2)C)=O)CN(C(c2csc(F)c2)=O)CC1C c1(C(=O)OC)sc(NC(=O)CCCC2(NC3CC(F)(CO)C3)CCC2)cc1C.C(C)(=O)C N1(C(C(C(CNC(COCC#C)=O)C)F)=O)CCC(C)(C)CC1C C=CCC(O)(CC=C)C(C)NC(=O)C(=O)NCC(=O)Nc1ccccc1CC CCCCS(=O)(=O)CC(=O)N(C(C)CN(C)C(c1cnc(C(=O)NC)cn1)=O)C c1(OC)cc(Br)c(F)cc1S(=O)(=O)NCc1ccc(C)cc1OC C(CCCCCN=c1ccnc[nH]1)N(C(CCC(=C)C)=O)C C1(C(=O)NC2CC(NC(c3cc(Cl)c(F)c(Cl)c3)=O)C2)CC2CCCCC2O1 C(=O)(C(CCC)C(C)C)N(CC(=O)NC(CC#C)CCOC)CCOC Cc1cc(C#N)cnc1C(N1CCCC1(C)C(=O)NC(C1CCCCC1)C)=O C1(C(=O)NC2C3CN(C(=O)CCSC(F)(F)F)CC23)CCC2(CCC2)C1 C(=O)(C(=O)C(C)(C)C)NC(C(=O)N(C)Cc1c[nH]nc1C)CC1CCC1 CC(C)(C)C(=O)CCCC(=O)N1CCN(C(=O)CC2CCC(=O)NC2=O)CC1 c1(C(=O)NC2C3CN(C(CSc4cccc(C)c4)=O)C2C3)cscc1S(C)(=O)=O C12(CNC(=O)Cc3cccnc3)CCCCC1N(C(c1ccc(F)cn1)=O)CC2 N1(C(C=CC)=O)CCN(C(c2cc(C)co2)=O)CC1C1CCCC1 c1(CC)ccccc1-n1cncn1.n12nncc1NC2=O c1(-c2c(C(N3CCC(C)(C(F)(F)F)C3)=O)c[nH]n2)nc2ccccc2s1 C(=O)(CCS(=O)(=O)CC(C)C)N1C2CN(C(c3c(C)cccc3Br)=O)CC1C2 C1(O)(CCNC(C2N(C)CCCC2)=O)CCCN(C(=O)C=C2CCOCC2)C1 CCC(CCC(=O)N1CC(=O)NCC1C(N)=O)NC(C1CC(C)N(C)C1)=O c1(OCC)cc2c(cc1Br)C(NCc1ccc(C)c(S(N)(=O)=O)c1)CCC2 N1(C(C=C(C)Cl)=O)C2CCC1CN(C(c1cc(O)c(F)cc1N)=O)C2 c1(OC)cccnc1NC(C1CC(O)CN1C(=O)CN1CCCC1)=O Cc1cc(Cl)c(C(=O)NCC2CCC(C)CN2C(c2cnsc2)=O)cc1F CCC(CNC(C1CCC1CNC(c1cc(N)cc(F)c1)=O)=O)(CC)CC c1(OC)c(C(N2CCC23CN(C(C2CCC(=O)O2)=O)C3)=O)cnc2ccccc12 c1(C2(C(=O)NCC3N(C(C(CC)N(C)C)=O)CCC3)CC2)cccc(OC)c1 N1(C(c2ccc(OCC)cc2)=O)CC2CN(C(c3[nH]c(=N)ccc3C)=O)CC2C1 c1(CC(N2C3CN(C(CCCCOC)=O)CC2C3)=O)c(C)nc2ncnn2c1C N1(C(c2c(CC)ncnc2)=O)CCC(O)C(NC(=O)C(C)C2CCCC2)C1 c1(OC)c(C(N2CC(CN(C)C(c3ncc(F)cc3F)=O)C2)=O)ccc(Cl)c1Cl c1(NC(=O)C(N2CCCC(NC(=O)C(F)(F)F)C2)=O)ccc(F)c(F)c1 C(c1ccsc1Br)=CC(=O)N(CC(C)NC(CCCOC(C)C)=O)C O=C(CC1=Cc2ccccc2C1)NC1CC1NC(c1cc2ccccn2n1)=O c1(C(=O)NC2C(NC(=O)CCCN3CCCCC3)C2)cnc2c(c1)CCC2 CCC(C)CCCC(=O)NC(C)C(CO)NC(c1cc(C)ncn1)=O c1(OC)ccc2c(C)cc(-c3cc4cc(C(=O)NC(C)C)ccc4s3)nc2c1 c1(C(=O)OC(c2cnc(N(C3CCCN3)CC)nc2)=O)cnc2cc(C)ccn12 c1(-c2cn(CC3N(Cc4cc(C(=O)O)oc4)CCC3)nn2)cnc(Cl)c(Cl)c1 N=c1ncc(C(=O)NCC2(O)CN(C(C3CCCC(O)C3)=O)C2)c[nH]1 c1(CNC(C23N(C(CC4CC(C)C4)=O)CCC2C3)=O)cc2cccnn2c1 C1(C(C)(C)NC(c2cc(C(C)C)[nH]n2)=O)CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1 C(=O)(CCC(C)S(C)(=O)=O)NCC1N(C(CC(C=C)(C)C)=O)CC2(CC2)C1 CC(C)C(CC(=O)NCC(C)(C)CN(C)C)NC(=O)C(N1CCOCC1)C CN1C(=O)NCC1C(=O)NCc1cn(CCNC(=O)COCC(F)F)nn1 C#Cc1cn(C)nc1C(=O)NC(C(=O)N1CC(NC(C)=O)C1)C1CCCC1 Cc1sccc1C(N1CC(OCCNC(C2CCCC2C)=O)C1)=O C1(NC(C2(SC)CC2)=O)CCN(c2ccnc(Cc3ccccc3)n2)CC1F C(=O)(CC(C)(C)COC)N(CC(C)NC(C1CCC(=O)NC1)=O)CC C(C(C)(C)C#CC(=O)NCc1cc(C)cnc1F)NC(C1C(=C)C1)=O c1(C(N2CCC(F)(CNC(=O)CC3CCCCN3)C2)=O)cc(Cl)ccc1Cl CN1CCC(n2nccc2-c2ccc(N)cn2)CC1.C1(=O)C=CCO1 c1(OC)nc(Cl)ccc1C(=O)NCCC1CCN(CC(=O)NCc2cccs2)C1 CC(C)(C)CCC(=O)NC1CCCC(NCc2ccccc2F)C1 c1(N2CCC(CNC(c3ccc4nn[nH]c4c3)=O)C2)ncnc2cnccc12 N1(C(CCNS(CC)(=O)=O)=O)CCCC(C)(C)C1CNC(C1CCCCC1(C)C)=O C1(NC(COCC(=C)C)=O)CCN(C(=O)C(C)(C)C2CCCO2)CC1(C)C C1(CC)CN(C(=O)C(C)(CC)CC)CCN1C(=O)CC(C)F N1(C(C2CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(O)C3)C(F)(F)C1 C(=O)(C(CC)CCCC)NC(CC#C)(C)C(=O)NCc1ccns1 c1(CC(N2CC(C)C(CNC(c3[nH][nH]c(=N)c3Br)=O)C2)=O)cnc2n1CCOC2 C(=O)(C1=CC2(CCOCC2)C1)N1CCC(NCCOC(C)C)CC1 C12(CC(N3CCC(COC)(NC(=O)C=C(C)C)CC3)=O)CCC(CC1)C2(C)C C12(C(N3C(CNC(C(c4cccs4)SC)=O)CC(O)C3)=O)CC(C)(C1)OC2(C)C c12cc3ccc(cc3[nH]1)OC2=O.C(CCCC1CCN1)N(CC)CC C(CC(C)CC)(C(=O)NCc1n[nH]c(CC)n1)NC(CC=C)=O c1(CNC(C2(F)CCCN(C(=O)CC3CC4CCC3C4)C2)=O)cc(F)cc(F)c1 N1(C(CCCC)=O)CCN2C(=O)C(NC(c3c[nH]c4nccc-4c3C)=O)CC2C1 C(N(C)N1CCCN(c2ccncc2)CC1)c1c(CC)onc1C c1(C(=O)NCC2CCC(CNC(CC=C=C)=O)CC2)ccc(F)c(CC)c1 c1(C(=O)NCc2cccs2)n[nH]c2c1CSCC2.C1(=O)COCCN1CCOC c1(C(=O)NCC(CNC(C(C2CCCO2)OC)=O)(C)C)c(F)cc(C)cc1F c1(OC)ncc(CN2CC(OC)CC2C(=O)OC(C)(C)C)cn1 C(=O)(C(C)P(C)(C)=O)NC(C)CCN(C)C(C1(c2ncccc2F)CCC1)=O c1(NC(=O)CC2CCC(NC(=O)C3=COCC3)C2)ncnc2ccsc12 n1(CCC)ccnc1CN(C(C1CCC(C)C1)C(=O)NCC(F)F)CC c1(C(=O)NCC(CO)NC(=O)C(O)CF)ccc2c(c1)OCC2 C#CCCCCC(=O)N(CCCNC(c1cc(C(=O)OC)no1)=O)C c1(C(N2CC(SC)C2)=O)ccnc(CNC(c2ccnc(CO)c2)=O)c1 C(=O)(C#CC1CCOCC1)N1CCC(NC(Cc2cc(C(C)C)no2)=O)CC1 C1(NC(=O)CC(F)F)CN(C(C2CC3CC3C2)=O)CCC1C(F)(F)F CC(C)C(C(=O)NCC(O)CNC(c1ccnnc1S)=O)NC(N)=O C(C(C)(C)CNC(=O)CC1CC=CCC1)NC(C(C1CCC1)OCC)=O N1(C(C2(CSC)CCC2)=O)CCC(CN(C(=O)C(C)CF)C)CC1 C1(C(=O)NCc2cnc(CC)s2)CC(F)(F)CN1C(=O)C(C)(O)C1CCC1 CCCCCCCC(=O)N1CCCC1(C)CNC(=O)Cn1ncnn1 n1(CCCC)ncc(C(N2CCCC2CCCNC(C2(C)C=CCC2)=O)=O)c1C CN1CCC(F)(CNC(C2CN(C(c3c[nH]cc3C3CC3)=O)CCO2)=O)C1 C1(O)(CC)CN(C(=O)C(CC2CCCC2)NC(=O)Cc2ccc[nH]2)C1 N1(Cc2scc(C)n2)CCC(C2CCCN(C(=O)Cc3cccc(Cl)c3)C2)C1 C1(C(N(C)CC2CCSC2)=O)C2CCN(C(C3CCCC(C)(C)C3)=O)CC12 C1(COC)(CNC(=O)CCc2ccn(C)n2)CN(C(=O)CCc2cn(C)nn2)C1 C1(C(N2CCC(OC)C2)=O)CC(O)CN1C(=O)CCCc1cccs1 N1(C(C(C2CCC2)OC)=O)CCC(N(CCO)C(c2cn(C3CCCC3)nn2)=O)C1 C1(C(=O)NCC(=O)N(C2CCN(CC(F)F)C2)C)CCOC1C(F)(F)F n1(CC)ccc(C(=O)NCC2COCC2NC(=O)C(c2ccc(F)cc2)F)c1C c1(CNC(=O)NCc2cnc3n2CCS3)c[nH]c2cccc(Cl)c12 N1(C(CC=CC)=O)CC(CNC(=O)CNc2cccs2)C(C)C1 c1(C(N(CCCNC)C)=O)coc(C(F)F)n1.C(=O)(CCOCC(F)F)N N1(C(c2ccsc2C(F)(F)F)=O)CCCC1C1CCCN1C(c1cnns1)=O C(=O)(CC(C)(C)CC(=O)NC(CCC(C)N(C)C)=O)N1CC2C(SC)(C2)C1 C(=O)(C1=CCCCCC1)NCC1C(NC(C(c2ccccc2)OC)=O)CCC1 c1(C(N2CC(CCCCNC(C(CC)F)=O)C2)=O)ccc(-c2cnn(C)c2)nc1 CC1(CNC(=O)C(F)(F)c2ncccn2)CC(NC(C2CCCCS2)=O)C1 N1(C(CCCOC)=O)CCN(C(=O)CSC(F)F)CC2CCCCC12 C1(NC(c2cc(CC)no2)=O)CN(C(C2CC3(CC3)CO2)=O)CC1C n1(C(C)C)cc(CNC(c2cnn3c2OCC3)=O)c(O)nc1=O C(C)(C)(CCC(=O)NC(C)C(=O)NCC1C2CCCCCC12)OC C1(C)(C(=O)NCCNC(C2CN(C(C(C)n3cccn3)=O)C2)=O)C=CCCC1 N1(C(C=C(CCC)C)=O)CC(C(=O)NCCC(=O)N(C)C2CC2)C(F)(F)C1 C1(SCC)CCC(C(=O)NCC2CC(NC(=O)C(n3cc(C)cn3)C)C2)CC1 CC1CC(c2nnnn2C)(NCC2(C(C)CCO)CCC2)CC1 c1(C(=O)NCCC2CCCN2C(C2CC(C(F)(F)F)C2)=O)ccn2ccccc12 c1(COC)nc2ccccn2c1C(=O)NCC1CCN1C(C12CC(O)C1C2)=O C1(NC(C(c2ccc(OC(C)=O)cc2)CC)=O)CCN(C(=O)CO)CC1O c1(CNC2CCC3C(CO)C32)ccc2nncn2c1 N1(C(c2cc(C)no2)=O)CCCC(CC(=O)NC(c2ccccc2)CF)CC1 CN1CCCCC(C(=O)N(CCCNC(C2CC(=C3CCC3)C2)=O)CCO)C1=O CC(C)CC(O)C(=O)NC(c1nc(C(=O)NCC2CCCC2CF)co1)C c1(OCC(=O)NCC(CNC(c2nscc2N)=O)OC)nn(C)cc1[N+](=O)[O-] CCC(C)(CCNC(=O)CC1SC(=N)NC1=O)NC(C1CCS(=O)(=O)C1)=O c1(C(=O)NC2CC(NC(C3CCOC3c3cn[nH]c3)=O)C2)cccc(C(F)F)c1 CCC(C(=O)N1CC(NC(C2CCCSC2)=O)C1)n1ccc(C2CC2)n1 c1(NCC2C(CC)CCOC2)ccc2nc(C)sc2c1 c1(Cn2c(C(=O)NCC(C)(C)Cc3ccccc3)ccn2)cccc(Cl)c1 c1(NC(=O)NCc2nnc(CO)s2)cc(N2CCCCC2)cc(Cl)c1 c1(C(N2CC(C(=O)OC)C(F)(F)CC2)=O)ccc(Br)c2ncccc12 C1(C(CC)C)CCC(CNC(=O)NC(C)C2CC2)CC1 N1(C(CCc2n[nH]c(=N)s2)=O)CCOC(CNC(C2CCCC2(F)F)=O)C1 C1(C(=O)NC(CSC)C(=O)NC(c2nc(=O)o[nH]2)C)CCCCC1CF C(CCCc1ccccc1)(C(=O)NC(C)CC)N(C(CC)C)CC(=O)OC C1(C(N2CC(c3nc(C)no3)C2)=O)(CNC(c2cnc(CC)s2)=O)CC12CCC2 C(=O)(CCC(=O)N1CCC(CCNC(c2cccc(CS(C)=O)c2)=O)C1)NCC C1(COC)CCCN(C(=O)C(C)NC(=O)CN(CC(C)C)C(C)=O)C1 c1(C(N(CC(C)NC(=O)Cn2nccc2C)CC)=O)ccc(C)c2ccccc12 C1(CCCNC(c2nc(CCC)sc2)=O)CCN(C(=O)Cc2cn[nH]c2)CC1 C(=O)(C1CCCc2nnn(C)c21)N1CCCC(N(C(=O)CCC(C)C)CC)CC1 N1(CC(=O)NCCC2(O)CCCN(C(CCC#CC)=O)C2)CCc2sccc2C1 Cc1nn(C)c(Br)c1C(N1CC(NC(c2ccc(O)c(Cl)n2)=O)C1)=O c1(C(=O)NCCC(=O)OCC(C)OC)ccc(OC2CC2)cc1 c1(C(N2C(C(=O)NCC3N(CC)CC3)C=CC2)=O)ncnc(O)c1F n1(CC)c(SC(=O)CC23CCCC2C3N=c2[nH][nH]cc2CO)nc2ccccc12 N1(C(C2(COC(C)C)CC2)=O)CCC(O)(CNC(c2cc(C)cc(O)n2)=O)CC1 N1(C(C2CC3CCC2O3)=O)CCC2(C1)CN(C(C1(F)CCOC1)=O)CCO2 c1(NC(c2c(F)cc(Br)cc2F)c2n(CCC)nnn2)ccc2nn[nH]c2c1 c1(CO)cn(Cc2conc2CC(N2CC(n3ccnn3)C2)=O)nn1 CCC(C(=O)N1CCN(C(=O)COC(F)(F)F)C(C2CCCC2)C1)C(C)(F)F Cc1cc2cc(C(=O)NCC3(O)CCN(C(=O)Cc4cnsc4)C3)c(Cl)cc2[nH]1 Cc1cccc(C(N2CCN(C(=O)CCF)C(C)C(C)C2)=O)c1[N+](=O)[O-] C(=O)(C(C)CCC(C)(C)C)NCC1(OC)CCN(C(=O)C(C)NC(N)=O)CC1 c1(CNC2C(CC#N)CCC2)ccc(I)c(F)c1F c1(CN(C(CCCNC(c2n(CC)ncn2)=O)=O)C)ccccc1O N1(CC2CCN(C(=O)NCc3nnc(C4CCC4)o3)C2)CCCOCC1 c1(C(=O)NCC(CNC(c2[nH]cc(C(=O)OC)c2)=O)OC)ncn2c1CCCC2 c1(N2C(CCNC(c3c(CC)ncs3)=O)CCC2)ncnc2c(Br)cccc12 N1(C(CC(CC)NC(=O)C(C)=NOCC#N)=O)CCN2C(=O)CCC2C1 N1(C(CNC(CC)=O)=O)CCC(C)(CNC(=O)C(N2CCSCC2)C)C1 C(C(C(=O)NC1CC(CC)C1)n1cc(CN2CCCC2)nn1)OCC C1(C(N2CC(C)N(C(c3ccnc(Cl)c3N)=O)CC2)=O)CCC2(C1)CC2(F)F c1(SC)cncc(C(N2CCC(N3CCN(NC(C4(C)CCC4)=O)CC3)C2)=O)c1 CS(=O)(=O)CCC(=O)NC12CCC(C(=O)NCC3CC(O)CCO3)(CC1)C2 C1(CC(=O)N(CCCC(=O)NCC(=C)Cl)C)C(C)(C)C1(C)C c1(C(N2CCCC(O)(CNC(Cn3c(C)cnc3)=O)C2)=O)ncnc2sccc12 c1(CC)ccc(CC(=O)N(C2CCCN(C(=O)CC3CCCO3)C2)CC)cc1F C1(C(=O)NC(CC)CO)CC(F)(F)CN1C(c1ccnc(C)n1)=O C1(C(=O)NC(C(=O)N(CC=C)CCO)C2CC2)CC(C)(C)CO1 Cc1ccc(C=CC(=O)NC(CNC(C2CCC(CO)CC2)=O)C2CCC2)nc1 Cn1cc(C(=O)N(CCC(C(C)(C)C)NC(=O)C=CC=C(Cl)Cl)C)n(C)c1=O C(=O)(C(CO)C(F)(F)F)NC(c1c(C(=O)NCC(C)N(C)C2CC2)con1)C N1(C(c2ncn(C(C)C)n2)=O)CCCN(C(c2coc(N(C)C)n2)=O)C(C)C1 c1(C(N(C)CC2CCCCN2C(c2cnc[nH]2)=O)=O)cc(F)c(F)cc1O C1(C(N2CCN(CCOC)CC2)=O)CCCCCN1C(=O)Cc1ccnn1C N1(C(C(C)NS(CCCC)(=O)=O)=O)CC2(CCN(C(=O)CN3CCOCC3)C2)C1 C1(NC(c2ccoc2)=O)CN(C(C2(CC(=O)OC)CC2)=O)CC(C)(C)C1 O(NC(=O)CCCCC(C)C)C(C(=O)NCC(COC)(F)F)CC(C)C c1(CN2CCC(C)(NC(c3c(C)cccc3)=O)C2)cccc2[nH]ncc12 C1(C(=O)NC(c2cn(C)nc2)C(=O)N2CC(N3CC(O)C3)C2)CC2(C1)CC(O)C2 c1(CNC(c2ccc(C(=O)OC)cc2F)=O)coc(S(N)(=O)=O)c1 c1(C(=O)NCCOC2CCN(C(c3c(C)n(C)nn3)=O)C2)cc(Cl)c(Cl)n1C Cc1cc(C(=O)NCC(O)CN(C(=O)C(C)NC(=O)OC(C)(C)C)C)cc(F)c1 C(=O)(C1COc2ccccc21)NC1CCCC(NC(c2cc(C)nc(O)c2)=O)C1 C(=O)(NNC(=O)OC(C)(C)C)NC1(c2n(C)ccn2)CC1 N1(C(c2noc(C)c2[N+](=O)[O-])=O)CC2CCN(C(=O)C=C3CCCC3)CC2C1 C(=O)(CCCC(C)=O)N1C(C)(CNC(CC2(CSC)CC2)=O)CCC1 N1(C(C2=C(C)OCC2)=O)CC2(CCCC2NC(c2cccnc2OC(F)F)=O)C1 C(=O)(CC(F)(F)C(C)C)N1CCC(CNC(C=Cc2c(C)noc2C)=O)C1C CCCC(C(O)C(=O)NC(CC)C1CC1)NC(c1cn(C)cn1)=O c1(NCCCC(C)NC(C2CC(c3ccncc3)C2)=O)cc(C(F)(F)F)ncn1 CC1(C)OCCC1CC(N1CC2C(CC(=O)NCC(C)(C)OCCO)C2C1)=O C(=O)(C1=CCCCC1C)NCC(CCC)C(=O)NCCC#CCO c1(N(C(C)C)CC2N(C(CC3CC(OCC)C3)=O)CCC2)ncc(C(F)F)cn1 C1(C(N(CCNC(c2cc(C)on2)=O)C)=O)CC2CCC(C1)N2c1cnccn1 c1(CC)ocnc1C(=O)NCCCC(C)NC(=O)CCCn1ccnc1 C=CCC(CC(C)C)C(=O)NCCCCCC(=O)N(CCSC)CC CCCCC(CC(=O)NCCCC(C)(C)OC)NC(=O)C1=NOCC1 C1(C)(C(=O)NCCC(CCC)C)CCN(C(=O)CC(CC)OC)CC1 C12(C(=O)NCC34OCC(NC(C=Cc5occ(C)n5)=O)(C3)C4)CCC(CC1O)C2 Cc1cc(CNC(=O)N(CCN(C)C)Cc2ccc(Br)cc2)c(C)cc1O C1(NC(c2cccc(CNC(=O)OC)c2)=O)CN(C(c2ccsc2)=O)CC12CC2 N1(CCc2cc(OC)cc(Br)c2)CCN2CCS(=O)(=O)CC2C1 C(C(C)(C)C(=O)N1CCC(OCCO)C1)N(C(CNC(C1C(C)C1)=O)=O)C C#CCCCCCC(=O)N1CC(NC(C2(C)CCN(C)C2)=O)CC12CCC2 c1(CC)cc(F)ccc1C(=O)NCCOC(C)(C)CNC(=O)Cn1cc(Cl)cn1 N1(C(C2N(N=O)CCC2)=O)CC2CC(C1)CN(C(=O)CCc1ccco1)C2 C(c1cccc(Br)c1)=CC(=O)NC(CNC(c1n(C=C)nnc1)=O)(C)CO C1(C(=O)NC(C2N(C(CCC(C)(F)F)=O)CCC2)(C)C)CC2COCC(C1)C2 c1(OCC)ccc(Br)c(C(F)(F)F)c1.c12cc(cc(F)c1)CNc1ccc-2nc1 Cc1ccc(NC2C(CO)CCN2C(c2ccc(Br)cc2)=O)c(-n2ccnn2)c1 c1(C(=O)NC(CNC(C=C(C)Cl)=O)CO)cncc2c1CCNC2=O C(=O)(CCCC(F)(F)CO)N1C(CCN(C(CCC(CC)OC)=O)C)CCCC1 Cc1cc(F)ncc1CN1CCOC(C(=O)Nc2ccc(Br)c(F)c2)C1 c1(C(=O)NC(C2CCOC2)CNC(C2(C(F)F)CC(=C)C2)=O)ncc(C)cc1C c1(C(=O)NC(C(C)NC(CN(CCC)C)=O)C(C)C)ccc(F)c(OC(F)F)c1 CC1OC2CCC1(CNC(Cc1ncns1)C(=O)O)C2 C#Cc1ccc(C(=O)NC2(C(=O)NCCCN3CCCC3)CCSC2)c(C)c1 C1(C(=O)OCCCN(CCC(=O)OC)CC(F)(F)F)CC2CCC1NC2=O N1(C(c2c(NCC)scn2)=O)C2CCC1C(CNC(c1cc(C3CC3)no1)=O)C2 CS(=O)(=O)c1cccnc1NCCCNC(=O)C(F)Oc1ccc(Br)cc1 c1(NC2(CC(=O)NC3C4CC5C3C5C4C(=O)NC)CCC2)cc(F)cc(F)c1 Cc1cccc2c(C(=O)NC3CCCC3NC(c3csc(C4CC4)n3)=O)c[nH]c12 C1(C(N(CC#C)CCO)=O)CCCO1.C(CCF)N(C(=O)C)CCC(C)CC n1(CCC(=O)NCCC2CCC(NC(CCOCC)=O)C2)cnc(C#N)n1 N1(CCOC)CC2(CCN(C(=O)CC3(C)CC(C)=NO3)CC2)OC1=O Cc1cc(F)ccc1CNCc1cn(-c2cccc(C#N)c2)nn1 CCC(C)C(CN(CC=CC(=O)NC(=O)CCCn1ccnc1)C)CO C=CC(C)CC(=O)N1CCCC1CNC(=O)C1=CSCS1 C1(C(=O)NC(C)CCNC(=O)CCCCCNC(N)=O)CS(=O)(=O)CC(=O)N1 Cn1c(C(N2CCCCC2C2CCN(C(C3CCCS3)=O)CC2)=O)nnc1S CC(C)CC(=O)C(=O)N(C(C)CCNC(=O)C(C)CCc1cccc(F)c1)C Cn1c(C(N2CC(C(=O)NC(CC3CC3)CO)C(F)C2)=O)cccc1=O c1(C(C(=O)NC)N(CCC)CCOC)n[nH]c2cc(OC)c(OC)cc12 N1(C(CC(C)C2CC2)=O)CCCC(O)(CNC(c2cnn3c2N(C)CC3)=O)CC1 C1(C(=O)NCCc2c(C)nn(C)c2)CCCCCN1C(C1C(C#N)C1(C)C)=O c1(C(=O)NCC(CNC(c2cncc(C)c2)=O)F)c(C)nc2sc(C)nn12 C1(NC(=O)C(=O)c2ccco2)CCC(c2ccccc2)C1 C1(C(=O)NCC2CCC(NC(c3c(CC)cccn3)=O)CC2)CC2(CCC2O)C1 N1(C(c2c(CNC(c3c(C)nc(CC)o3)=O)nnn2C)=O)CCC(C)CC1CC C1(C(=O)NCc2c(C(N(C)CC3(O)CCOC3)=O)n(C)nc2)CC(=O)OC1(C)C Cc1nn(C)c(C)c1C(=O)NCC1(F)CCCN(C(=O)CC2C=CS(=O)(=O)C2)C1 CC(F)(F)C(F)C(=O)NCC1CCN(C(=O)C(C)(O)C2CCC2)CC1 N1(C(C2C(C)CCC2)=O)CCN(C(C2CCC(NC(N)=O)CC2)=O)CC(O)C1 C(c1csc(C(F)(F)F)c1)=CC(=O)NCC(C)(C)NC(C(C)NC(COC)=O)=O c1(C(N2CCCC(CCNC(C(C(C)O)(F)F)=O)C2)=O)cc2c(cc1N)CCC2 N1(C(C2(OC)CC2)=O)CCC(C(C)NC(=O)Cc2csc(-c3csc(C)n3)n2)C1 CC(C)(CCCNC(c1coc2c1COC2)=O)C(=O)NCC(C)(O)C1CCC1 N1(C(c2c(C(C)(C)C)ccc(N)c2)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)C2)C1 C1(CN(C(C(N2CCOCC2)C)=O)C)COCCN1C(C1CCCN1C1CC1)=O C1(C#CC(=O)N(C(c2cccc(Cl)c2)=O)CC2CCCC2)(CN)CC1 c1(C(C(=O)NCC2(CO)CC2)N(C2CCCC2)C)ccn2ncc(Br)c2c1 CC1CN(C(=O)CC2CCC(O)C2)CCC1CNC(c1cc(C(N)=O)[nH]n1)=O C(=O)(C1=NOC(C)(C)C1)N1C(C(=O)NCC2(CC)CCOC2)CCCC1 N12CCCCC1C1CCN(C1)CC2=O.Cc1ccoc1NC(=O)C=CC=C(C)C N1(C(c2c(CCC)[nH]cc2)=O)C2CCC1CN(C(c1cnc(C(C)C)n1C)=O)C2 c1(-c2ccc(C(N(C)C)=O)cc2)ccn2ncc(C(=O)NCCC(C)(C)O)c2c1 CC(C)C(O)CC(=O)N1CCC(NC(=O)CCCc2cccnc2)C1C C(CC(C)(C)CN=C(NCC(C)(C)C#N)NCC(C)(C)C)SC CC1(C(=O)NCC2(CNC(=O)C(F)(F)c3ccccc3)CC2)CC=CCC1 c1(N(C)C)cc2c(cn1)CN(C1CCNOC1)CC2 Cc1c(-c2nc(CC(=O)Nc3cccc(F)c3)no2)ccn1C c1(C(N)=O)cc(COC(C2Cc3cc(Br)ccc3O2)=O)c2n1CCCC2 CS(=O)c1cccc(C(=O)NCc2ccccc2CNC(c2ccncc2)=O)c1 Cc1cnc(Cl)[nH]c1=NC1CCCOC1C1CCN(C(=O)CC2(C)CC2)CC1 C1(CC2N(Cc3ccn(C)c3)CCC2)CCN(C(c2cncnc2)=O)CC1 Cc1cncc(C(=O)N(CC(C)O)CCNC(c2ncc(F)cn2)=O)c1Cl C(=O)(C1CCCc2c1ncn2C)N1CC(O)(CNC(c2n(CC)cc(Cl)c2)=O)C1 S(=O)(=O)(CC(=O)NCC1CCN(C(c2ccc(NC(C)=O)s2)=O)C1)NC c1(C(=O)NC(CNC(C2CCN(CC)C2)=O)C(C)C)cncn(C)c1=O N1(C(C(C=C)(C)CC)=O)CC2(CCCCN(C(=O)CC(C3CCC3)C3CC3)C2)C1 Cc1nc(CC(=O)NC(C)(CNC(=O)CC(O)C2CCCC2)C2CC2)co1 C1(NC(CC=C)=O)CC12CCN(C(C1CCCOCC1)=O)C2 C1(NC(C(C)C2CCCC2)=O)CN(C(=O)Cc2ccc(Cl)cc2)CCC1(C)C N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)CCC(=O)NC)CC(C)C1 C1(C(N2C(CNC(C3N(CC)CC3)=O)CCCC2)=O)CC2(CCCO2)C1 C1(NC(C(C)N(C(c2coc(C(F)F)c2)=O)C2CC2)=O)CC(C)N(C)CC1C C1(C(=O)OC)CCN(CC(=O)N(CCN(C)C)Cc2cccc(C)c2)C1C N1(C(C2CC3(C2)CC3F)=O)CCCC1(C)CN.c1(C(C)=O)ccc(C(=O)NC)o1 C(=O)(C(C)(F)C(F)(F)F)NCCCC(C)NC(=O)Cc1ccccc1Br C1(NC(C2C(NC(=O)C(O)C3CCCC3)CCCC2)=O)CCCC(C2CC2)C1 n1(C(C)C(=O)NC(C)(CNC(c2cnn(CCO)c2)=O)C2CC2)cnc(C#N)n1 C1(CNC(CCOCCC)=O)CCCCN1C(=O)C(=Cc1c[nH]cn1)F c1(OC)ccc(O)c(NC(C2(F)CCN(Cc3c(OC)cccc3C)C2)=O)c1 n1(C(CC)C)nc(C(=O)NCC(C(C)C)NC(c2ccc(C)s2)=O)cc1C c1(C(N2CC(CC)N(C(=O)C(O)C(C)(C)C)CC2)=O)cc(OC)cc(C#N)c1 N1(C(CC(=O)OC)=O)CC2CCC(C1)N2C(=O)CC1CC1C(F)(F)F C(=O)(C(F)(F)C(C)(C)O)NCC(CCC)NC(=O)CCC12CCC(CC1)C2 C(=O)(C(O)CC(N)=O)N(C(C(N1CC(C)(COC)C1)=O)(C)C1CC1)C c1(C(CNC(=O)NC2(CCC=C)CC2)N(C)C)cn[nH]c1 C1(OC)CN(C(c2sccc2-c2cn[nH]c2)=O)CC1NC(=O)CCF CC1=C(C(=O)NCC=CCNC(c2c(OC(F)F)cccc2Cl)=O)CCCC1 N1(CCCCCCC)CC2(CC(NC(=O)Cc3c(C)ncnc3C)CO2)C1 c1(C(=O)NC2C(CNC(c3cc(Cl)cs3)=O)CCCC2)cncc2c1CCC2 c1(NC(c2c(NC(=O)CCc3cc(F)ccn3)c[nH]n2)=O)cc(F)c(Br)cc1F c1(C2C(NCc3n[nH]c(-c4cccc(C)c4)n3)C2)ccc2c(c1)OCO2 CS(=O)(=O)C1CN(C(=O)CC2=CCCC2)CC1NC(=O)C(O)c1ccco1 N1(C(C2CCCN(CC)C2)=O)CCC(NC(=O)CC2COCC2O)C(CO)CC1 c1(C(=O)OC(c2ccco2)C)ccc(Br)c(NC(=O)CN(c2ccccc2)C)c1 C(C(CNC(C1(C)CC(C(F)(F)F)C1)=O)CO)NC(C1CC(C)C1)=O Cc1noc(C(C)C)c1C(=O)N(C)CC1(NC(C2(C(C)(C)O)CCC2)=O)CC1 c1(C(=O)NCc2c(C3CN(C(C4CN(C)C4)=O)C3)ocn2)ccc(F)cc1Cl C(=O)(C1CCCc2cccnc21)N(C1CCN(c2cc(C(N)=O)nc(Cl)n2)C1)C Cc1nc(Cl)c(NC2C(F)(F)C23CC3)nc1C N#CC1=C(C(=O)N2CC3CC2CCN3C(c2nncc3c2CCCC3)=O)CCC1 Cc1cc(C(=O)NC2CCCC(NC(c3cccc(Br)c3Cl)=O)C2)cc(C)n1 c1(C(=O)NCC(C)N(C(CCCOC(C)=O)=O)C)cc(OC(F)(F)F)ccn1 c1(C(=O)NCC(=O)OC)ccc(NNC(=O)C2CCC(C#N)C2)cc1 N1(C(CC(C)F)=O)CC2CCCC(CNC(c3ccnc4c3CCO4)=O)C2C1 C1(CC(N2CCC(Cc3cn(C4CC(O)C4)nn3)CC2)=O)SC2=NCCN2C1=O CC(C)C(C)S(=O)(=O)N=c1cc(CCCNC(N)=O)n(C)[nH]1 N1(CC(C)CF)CCc2cc(OCC3CC3)ccc2C1 N1(C(CC2(C)CC2(F)Cl)=O)CCN(C(=O)COC2(C)CCCC2)C(CCO)C1 Cc1cc(C(N2CC(N3CC(NC(=O)C=Cc4cc[nH]n4)CC3=O)C2)=O)c(C)o1 C1(C(C)NCCC=CBr)(OC)CCOC1 O=C1CCc2cccc(C(=O)NCC(CO)NC(=O)C(O)C(F)F)c2N1 c1(C(=O)NC2CCCC(NC(c3c(C)cc[nH]3)=O)C2)ccc(O)cc1F c1(C(C)NC(C2CCN2C(c2cn(C)cn2)=O)=O)c(N2CCCC2)cccc1Cl c1(CC(N2CCC(c3cn(Cc4cocc4CO)nn3)C2)=O)ccc(O)nc1 C1(O)(C(C)NC(c2scc(OC)c2)=O)CCN(C(=O)CN2C(C)CCC2C)CC1 CN1C(=O)Cc2cc(NC(=O)NC3CCC(F)C3)ccc21 N1(C(C(=O)N(CCOC)CC)=O)CCOCC12COCCN(C(C1CCCO1)=O)C2 c1(C(N2CC(C(C)NC(c3c(C)nc(O)cc3)=O)C2)=O)c([N+](=O)[O-])cnn1C C(=O)(C(CC(F)F)NC(=O)CC1CCCC1)NCC1CCN(C)C1 CC(C)CC(C)CC(C)C(=O)Nc1cncc(-c2cn(CCOC3CCC3)nn2)c1 C=C1CC(C(=O)NCC(CO)OC)(CNC(=O)C(O)CC)C1 c1(CC(=O)NCC(CNC(CCc2onc(C(C)C)n2)=O)C)c(O)ncnc1O CC1CCCC(CCNC(=O)C(n2cc(-c3ccccc3)nn2)C)C1 Cc1noc(C)c1CN(C)C(C1CC(CCNC(C2CC2Cl)=O)C1)=O c1(C(=O)NC(c2ccc(Br)nn2)C)ccccc1-c1ccc(C(F)(F)F)cc1 C(=O)(CCC(F)(F)F)N(C)CC1CCCCN1C(c1nc(Cl)c(Cl)s1)=O C1(C(=O)NCC2C3CN(C(C(CC)CC(C)C)=O)C2C3)CCc2nc(C)cn2C1 N1(C(CC2CCC(C#N)C2)=O)C2CCC1CC(C(=O)NC1CC3(CC3)C1)C2 C1(C(=O)NCC(C(=O)OC)C)CCN(C(C2CC3CCCC3C2)=O)CC1C C1(C(N(C)Cc2cncn2C)=O)CCC2(CC2)N1C(=O)C#CC1CC1 c1(OC2C3CN(C(c4cn5cc(C)nc5s4)=O)C(C3)C2)cnc2c(ccn2C)c1 CCCCCCC(=O)N(C)CC1CCN(C(c2cnc(C(C)=O)s2)=O)C1 C12(CNC(=O)Cc3csc(C(F)(F)F)n3)CC1CN(C(C1CC13CCCC3)=O)C2 Cc1ccc(C(N2CC3CC(NC(c4sc(O)nc4C)=O)C2C3)=O)cc1C#N C(CC(C(=O)NC1CCCC1CN(C)C)NC(=O)C1=CCSC1)=CC c1(CC)c(C(=O)NCC(O)CNC(=O)CCc2cccn2C)cnn1CC S(=O)(=O)(c1c[nH]c2nc(F)ccc12)NCCCN1C2(CCCS(=O)(=O)C2)CC1 C1(NC(CCCSC)=O)CN(C(C2(O)CCSCC2)=O)CCC12CCC2 c1(CNC2(c3n(CC)nnn3)CC(CC(C)C)C2)ncc(F)cc1F Cc1cccnc1CC(N)C(=O)NC1CCCC(N(C)C)C1 C#Cc1cc(C(N2CC(NC(=O)C(C)(C)OCC)C(C)C2)=O)cc(Br)c1 N1(C(COCC)=O)CC2CC2(C(=O)Nc2c(-c3ccccc3)noc2C(N)=O)C1 Cc1ccccc1C=CC(N1CCC(OCCNC(=O)C2=C(Cl)CC2)C1)=O C(=O)(CCCC(=O)NCC1(C)CCCN1C(C1CC1C(N)=O)=O)NCCC c1(C(=O)OC)nc(C(=O)NCC2CC2NC(=O)Cc2csc(C)n2)cs1 c1(CC(=O)Nc2c(C(N3CCC(=C)CC3)=O)scc2)ccc(F)cc1Br C1(NC(c2c(C)scc2)=O)CCC(C)(CNC(C2CC2C2CC2)=O)CC1 Cc1ccc(-n2ccnc2)c(C(=O)OCC(=O)NCCC2CC(=O)N(C)C2)c1 C1(N)C(=O)C1CC.C(C)(C(=O)N(CCO)CCN(C)C)OCCCC CC(C)(C)C(C)(C)C(=O)N1CCCC(NC(=O)CN2CCCNC2=O)C1 Cn1ccc2cc(NC(=O)NCC(c3ccc(O)cc3)O)ccc2c1=O Cc1cc(OCC(=O)NC2CCCCN(C(=O)CC3C=CCC3)C2)c(C)c(C)c1 N1(C(CCCc2ncc(C)o2)=O)CC(NC(c2sccc2C(C)C)=O)CC(C)C1 C#Cc1ccc(F)c(C(=O)N(C(C)CCNC(c2cncc3c2CCC3)=O)C)c1 C=CCC(CNC(c1ccc(C)cc1)=O)C(=O)NCCN(CCCC)C N1(C(=O)C(CO)C(F)(F)F)CCC(C2CCN(C(C3CCCOC3)=O)CC2)CC1 C#CCCCC(=O)NCC(C)(O)CNC(=O)C(C)(C)NS(C)(=O)=O c1(C(N2CCC(CC=C)(NC(C3CC(C)(O)C3)=O)C2)=O)ccc(OCC)cc1Cl c1(C(N2CC(OC)C(NC(=O)C(C3CCCCC3)F)C2)=O)nnn2c1COCC2 C1(C)(CNC(C2N(CC)CC2)=O)CCN(C(c2nocc2C(=O)OC)=O)C1 C(=O)(C1Cc2ccc(F)cc21)NCC1C(CNC(CCCC(C)(C)C)=O)C1 C(CCCOC)(C(=O)N(Cc1ccccc1)OC)NC(C(CCC)C#N)=O C(=O)(C(C(C)C)C(C)C)N1CC(C)(C(N2CC(C)CC(OC)C2)=O)C1 O=C(CCC(=O)C1CC1)NC1CC(CO)N(C(C2CC=CCO2)=O)C1 CC(C)CC(C)CN=c1nc(N(CCC(F)(F)F)C)c2c([nH]1)COC2 CCC(CNC(=O)Nc1cccnc1-n1ccnc1)C(C)C n1(CC)cc(C(=O)NCCn2cc(C(N3CCC(C(F)F)C3)=O)cn2)nn1 Cc1ccccc1CCC(=O)NCC1(C(N)=O)CN(C(=O)C(F)F)C1 N1(C(CC(CC)C2CC2)=O)CCOC2(CCCN(C(C3CCc4cncn4C3)=O)C2)C1 C(C(C)(COC)C(=O)NC(C)Cc1cn(Cc2nc(C(=O)O)cs2)nn1)OC N1(C(CCC)=O)CCN(Cc2ccccc2)CC1.C12CCC(CC1)NC2=O C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC1CN(C(CC(C)C)=O)CC1(C)C N1(C(CCCNC(C)C(=O)Oc2cc(Br)cn2C)=O)CCc2ccccc21 N1(C(c2ccc(C#C)cc2)=O)CCC2(CC(NC(c3cc(Cl)n(C)n3)=O)CO2)C1 C1(C(=O)NC(C)CC2CN(C(c3cn(C(C)(C)C)cn3)=O)C2)CCCCC1O C1(CCC)C(C)CCCN1C(C1(C(=O)NCc2cc(CC)n[nH]2)CC1)=O Cc1cc(C(N2CCOCC2CNC(=O)C(C)CS(C)(=O)=O)=O)cc2ccoc12 N1(C(C2C3N(C(C4C(OC)CCC4)=O)C(CC3)C2)=O)CCc2oc(C)nc2C1 C=CC1(C(=O)NCCOC(C)(C)CNC(=O)C(F)C(F)(F)F)CCCCC1 C(CCSC)(C(=O)NC1CCCN(C(c2n[nH]cc2Br)=O)C1)OC CN1CCN(C(=O)Cn2ncnn2)C(C(=O)NC2(CO)CC2)C1 C1(CC)CCCC1(C)C(=O)N(CC(C)(C)CNC(c1ccc(C(F)F)cc1)=O)C c1(NC(c2c[nH]c(Br)c2)=O)ccc(C2CN(C(=O)C(F)F)C2)cc1 c1(C(=O)NCCOC2(C)CCOCC2)coc2c1CN(C(=O)C(C)(O)C1CC1)C2 N1(C(c2nnn(C)n2)=O)CCN(C(=O)C(c2ccccc2Cl)O)CC1CCO Fc1cccc2c(CNCc3cc(Br)c4[nH]ncc4c3)c[nH]c12 C(C)(N=c1nc(Cl)[nH]c(C)c1C#N)C1N(C(C2=CC(C)(CC)C2)=O)CCCC1 c1(C(N2CC(C3(NC(CC4CN(C(C)=O)C4)=O)CC3)C2)=O)cn(C)c2ccccc12 c1(C(=O)NC23CN(C(CN(CCOC)C)=O)C(CC2)C3)cc(C)c(F)cc1F CCCCCC(CC)C(=O)NC(CNC(=O)Cc1cc[nH]n1)CC c1(CC(=O)NCC(CO)NC(c2cc[n+]([O-])cc2)=O)ccc2nsnc2c1 c1(C(N(C(C(=O)N(C(c2cnnn2C)C)C)C)C)=O)ccc(C2CC2)cc1 c1(SC)ccc(Cl)c(C(=O)NCC2(CNC(C3(C#N)CC3)=O)CC2(F)F)c1 N12C(CC3COCC13)CNC2=O.N(C1CC1)CC.C(C)(=O)N C(=O)(CCCC(F)F)N1CC2C(CNC(C3CN(C(C)C4CC4)C(=O)C3)=O)C2C1 c1(CS(=O)(=O)NC(c2ccc(F)cc2)C)ccc(Br)cc1F CC1CC2(CCCC2)CN1C(=O)C(C1CCN(C(C23CCCC2C3)=O)CC1)C N1(C(Cc2cc(C)ncc2)=O)CCC(O)(C(=O)NCC2CCOC2)CC1 c1(OC)cc(Br)cc(NC(N2CCN(C3CC3)CC2)=O)c1OC C1(CC(=O)NCC(CC=C)NC(c2ccnc(O)c2)=O)CC2(CCOCC2)CO1 C1(CC)(COC)NC(=O)N(CC(=O)NCC2CN(C(=O)CSC)CCC2C)C1=O Cc1[nH]nc2ccc(C(N3CC(CNC(c4coc(CO)c4)=O)CC3C)=O)cc12 N1(C(CC2CN(C)C2)=O)C2CCCC1CN(C(c1ccnc3ccncc13)=O)C2 n1(CC)ncc(C(=O)NCC2(NC(=O)C(O)C3CCCC3)CCCCC2)c1Cl c1(C(N(CC(CNC(CC(C)N(C)C)=O)O)C)=O)cc(F)c(Cl)cc1F N1(C(c2csc(C)c2N)=O)CCC2(CC1)CC2CNC(C1(CN(C)C)CC1)=O N1(c2[nH]c(=NCCOCC)c(C(N)=O)cn2)CCc2cccc(C(=O)OC)c2C1 N1(C(CCCCC)=O)CC2CCCC2(CNC(=O)C2=COCCC2)C1 CCC(CC)CC(F)C(=O)NC12CC(NC(c3cc(C(C)C)no3)=O)(C1)C2 c1(NC(C=Cc2n(CC)ncc2)=O)cccc(S(=O)(=O)N(C)C)c1 C(=O)(C(C)(Cl)Cl)NCCC1(C(=O)NC)CCC1.C12(CC1)C(=O)N2 C1(NC(C(CSC)OC)=O)CN(C(=O)Cc2c(C(F)(F)F)coc2C)CC1O N1(C(c2ccc(OCC)cc2)=O)CCCN(C(c2ccon2)=O)C(CO)C1 n1(CC(=O)NCC2(C(C)NC(C(C)OC)=O)CC2)cnc2c1CCCC2 c1(C(=O)NCCC(CNC(c2ncc(OC)cc2F)=O)O)c[nH]c(C)c(Cl)c1=O N1(C(c2c(NC(C)=O)cccc2)=O)CC(C(=O)NC(C)(C)CO)CC12CCOCC2 C1(NC(C2CC(OCC)C2)=O)CN(C(=O)CCCC(C)=O)C2(CCOCC2)C1 N1(C(C=COCC)=O)C2CCC1CC(CNC(=O)CC1COC(C)(C)CO1)C2 CCCCC(C(C(=O)O)NC(=O)NCc1ccc(C)cc1)Nc1nc(C(C)C)no1 CCCCCC(CC)C(=O)NCC1(NC(=O)CCNC(C2CCC2)=O)CCCC1 c1(CSC2(C(=O)NCC(C(C)C)NC(CCSC)=O)CC2)cccc(Cl)c1 CC1CC(C)N(C(c2cnccc2Cl)=O)CCN1C(=O)Cc1cnns1 C1(NC(C(n2cc(CCOC(C)=O)nn2)C)=O)CCSC(C)C1 c1(C(N(C2CCN(C(CC3CN(C)CC3O)=O)C2)C)=O)ccnc2c1CCO2 c1(C(N2CCC(C(C)NC(C3CC=CC3)=O)C2)=O)cc2cc(Br)cn2c(O)n1 C(CS(=O)(=O)NCC1CCC(c2cccc(C)c2)O1)(C1CC1)OC C1(C(N(CCCN(C)C(c2ccncc2)=O)C)=O)CCCC(=O)N1 c1(CN(CCC)Cc2ccccc2C(F)(F)F)ccc(C(=O)OC(C)C)cc1 c1(Oc2cccc(C)c2)ccc(Cl)c(NCC(=O)NCC(F)F)c1 c1(C(N2C(CCOC)CC2)=O)cc(OC)c(O)c(C(C)C)c1.C1(C(=O)NC)(OC)CC1 CCCC(CC(=O)NCCN1CC2CC2C1)NC(=O)Cn1cc(Cl)cn1 C1(C(N(C2CCN(C(=O)C=C3CCOCC3)CC2)CC#C)=O)COCC(C)O1 Cc1ccc(C(N2CCN(CC(N3CCC(C)(CN(C)C)C3)=O)CC2)=O)cn1 CC(C)(C)CCC(=O)NC1CCCC(Nc2cc(O)nc(O)n2)C1 C1(CC#C)(C(=O)NCC(C)Nc2nccc(CC#N)n2)CC=CCC1 C(=O)(C1=CCCSC1)NC(C1CCN(C(c2ccc(C(=O)OC)s2)=O)CC1)C CC1CC2CN(C(=O)C3=CC(C)(CO)C3)CC12.C12(CF)CCN(C1)C2=O c1(CNC(C2CCCO2)C#C)csc(NC(C)=O)n1 c1(C(=O)N(c2ncnc3c2CCCC3)C2CCNC2)cc2c3c(c1)CCCN3CCC2 c1(C(=O)NCC(C)(CO)NC(c2ccnc(CO)c2)=O)ccn2nnnc2c1 N1(C(c2sc(C)c(Br)c2C)=O)CC2CN(C)C(CO)C2C1 O=C(CCCSc1ccncc1)NCC1C=CC(NC(=O)C(O)c2ccsc2)C1 C1(NC(C=CC(=O)NC(C2CCCCN2C(C)=O)C)=O)CCc2c(n[nH]c2C)C1 O=C1CCCN(C(C2C3CC2N(C(=O)C=Cc2cncs2)C3)=O)C1CCO N1(C(C2(CC(=O)OC)CCCC2)=O)CC(n2cc(CCO)nn2)C(C)C1 c1(C(=O)NC2(CC)CCCN(C(C(CC)OC)=O)C2)cc(F)c(F)cc1Cl N1(C(C(CC(N)=O)O)=O)CC(O)(C2(CNC(=O)CCn3ccnn3)CC2)C1 CC(CC(=O)N(C1CCOC1)C(CC(=O)OC(C)(C)C)=O)CC(F)(F)F c1(C(N(C2CC3CC2N(C(C2CC2[N+](=O)[O-])=O)C3)C)=O)cc(F)cc(Cl)c1 N1(C(C(C)OC2CCCC2)=O)CCC(CNC(c2ccnn2C(C)(C)C)=O)CC1 c1(C(N2CCCC2)C)ccc(=O)n(CC(C)O)c1.C12(CC1)NC(=O)NC2 Cc1ccc(F)c(C(N2CC(C)CC2C(=O)NC2(C)CCCCC2C)=O)n1 CN(C)S(=O)(=O)NCC(=O)NC1CC(NC(=O)CC2CC3(CC3)CO2)C1 c1(C(c2n(CC)nnn2)NCC2CSCCO2)ccc(CC2CCCC2)cc1 CCCC(O)CC(=O)NCC1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CCOCC1 CC(C)CC(C#N)C(=O)N1CCC(NC(c2cc3c[nH]cnc-3n2)=O)C(F)C1 C1(C(N(CCCNC(C23CCCC2C3)=O)CCC)=O)CCN(OC)CC1 C=CC(C)(CCOC)C(=O)NCCN(C(=O)COCc1nnc(C)s1)C1CC1 CC1c2ccc(Br)cc2CCN1C(=O)NC1(S(C)(=O)=O)CC1 c1(C(=O)NC(CCCC)CNC(C2(OC)CCC2)=O)cc(Cl)c(OC)cc1C C(=O)(C(O)C(C)(C)C)NC12CN(C(CSc3nc(C)c(C(=O)O)s3)=O)C(C1)C2 C1(CCC2N(C(C3(OC)CC3)=O)CCC2)CCN(C(C2(C)CCCS2)=O)CC1 CC(N=c1ccc(Br)c(S(=O)(=O)N2CCCC(C(F)F)C2)[nH]1)C1CC1 c1(C(=O)NCC2(CO)CCN(C(CC3C(C)C3)=O)CC2)cc2cccnc2o1 CC1CC(NC(=O)Cc2nc[nH]n2)CCN1C(c1ccc(C2(O)COC2)cc1)=O C1(CC)CN(C(c2cnc(C)cc2Cl)=O)CCC1NC(C1(C)CCNC1=O)=O c1(CC(=O)NC2CC3CC(NC(C(CC)C)=O)C2C3)cc(F)c(F)cc1F Cn1cc(C(N2CC3CC(NC(=O)CO)C2C3)=O)n2cncc2c1=O CCC(CC(F)(F)F)C(=O)N(CC(C)N(C(=O)CCN(CC(F)(F)F)C)C)C c1(C(=O)NCc2cc(C(N3C(CC=C)CCCC3)=O)no2)ccc(O)c(CO)c1 N1(C(C2C=CCN2C(=O)Cc2ccns2)=O)Cc2ncsc2C1 c1(OCC)nc(C)ccc1C(=O)NCCC1CCCN1C(c1cnc(OC)s1)=O C1(C(=O)NCC2C(NC(Cc3ccc(C)nc3)=O)CC2)CCCCC1C1CC1 c1(C(=O)NC)ccc(C(=O)NC(C)CC(C)NC(=O)CC2CCCCO2)cn1 N1(C(c2[nH]cc(C#N)c2)=O)C2CCCC1CN(C(c1ccnc(O)c1)=O)CC2 C(=O)(C(O)CC(C)C)N1C(C(C(=O)NC(CC=C)C(=O)OCC)(C)C)CCC1 C(=O)(CC(=O)NC1CC1)N(CC(C)NC(C1CC=CC1)=O)C N1(C(C(C)(C2(C)CC2)NC(C)=O)=O)CCC(C)(C)C(NC(c2ccc(CO)o2)=O)C1 c1(C(=O)NCC2CCCN(C(CC)C)C2)ccccc1[N+](=O)[O-] C1(C(N(CC(C)C(F)(F)F)C)=O)CC12CCN(C(=O)Cc1cccc(F)c1)CC2 c1(C(C)=O)ccc(C(=O)N(C2CC(NC(C3CC3CF)=O)C2)C)nn1 c1(C(=O)NC2CC(CN(C)C)C2)ccc(-n2ccnc2)cc1 c1(C(=O)NC2CN(C(C(C(=C)C)(C)C)=O)CC2O)cc2nc(Cl)ccc2s1 Cc1nc(C#N)c(NCCC(=O)NCC2(NC(=O)Cc3ncc(C)s3)CCC2)o1 c1(CC(=O)NC2CN(C(c3cnc(O)s3)=O)CC23CC3)ccc(Cl)c(Cl)c1 C1(C(C)C)(CC)CCN(CCNC(=O)C2CC2)C1.c12ccc(s1)C2.c1(=O)c(=O)[nH]1 CC(C(=O)N1CC=CC1(C)C(N1CCCN(C2CC2)CC1)=O)S(N)(=O)=O C1(NC(c2nc(C)oc2)=O)CC2(C(=O)N(C)CC3CCC(C)CC3)COC1C2 c1(SCC)cccnc1C(N1CC2CC2(NC(C2CCCC3CC23)=O)C1)=O C1(C(=O)NC2(CNC(CCN(C)CCO)=O)CC2)CC2(C1)CC21CCC1 CC1CN(C(c2cnc(O)n2C)=O)CC1NC(c1cnn(C)c1Cl)=O C(N=c1cc(C)[nH]c(=NCCCN2CCCS2(=O)=O)[nH]1)C1CCC(COC)O1 C(=O)(C1=C(Cl)CCC1)N1CC(C(C)NC(=O)C(Cl)=CCl)OCC1 N1(C(C(C)n2ccnn2)=O)CCCC(O)(CN)CC1.C1(C(=O)NC)CC12CC2 N1(C(CCC#C)=O)CCC(C)C(NC(c2ccc(OCCO)cc2)=O)C1 c1(C(N2CCC(F)(CNC(C3(OC(C)=O)CC3)=O)C2)=O)ccc2ccoc2c1 N1(C(c2n(CC)c(O)nc2)=O)CC(CNC(=O)C(C)C(C)(C)C)C2(CC2)C1 c1(C(C(N2CCCC(N(C)C)C2)=O)OC)cc(F)ccc1F.C1(C)C(=O)O1 N1(C(COCCCCC)=O)CCC(C(F)F)(CNC(c2cn(CCO)nn2)=O)C1 C1(CCOC)CN(C(=O)C(=Cc2ccco2)C)CCN1C(=O)CCC1CCCO1 N1(C(CN2CC(=O)NCC2)=O)CC2CCN(C(C3(Cl)CC3(F)F)=O)CC12 C(=O)(CCP(C)(C)=O)N(CC(N1CCC(CCC2N(C)CCC2)CC1)=O)COC c1(C(N(CC(=O)NCC(CC)O)C(C)C)=O)cc(C(C)=O)c[nH]1 C1(C(=O)Nc2n[nH]c(C(F)(F)F)n2)CN(C(c2ccns2)=O)CCC1(F)F C1(NC(c2c(CC)csc2)=O)CC(F)CN(C(=O)C(Br)=C(C)C)C1 C1(C(=O)NC2(C)CCCN(C(c3n(CC)ncc3Cl)=O)C2)Cc2nc(C)cn2C1 C(CCCC(C)NC(=O)C(CCC)OCc1ccccc1)NC(CCC#C)=O CC1CC(c2ccccc2)N(C(=O)C(=O)NC2CC2C2CC2C)C1 N1(C(C(CC)N(C)C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 C[S+](C)CCC(O)C(=O)N1CCCCC1CNC(C1CCCN1C(N)=O)=O c1(C(C)(C)NC(c2nc(CCC)oc2)=O)ccc(OC(C)C)cc1 CCC(C(=O)N1C(C(=O)NCCCCC2CC2)CC1C)Oc1ccccc1 C1(C(=O)NCC(NOC)=O)CC(F)CCN1C(C1CC(O)CN1C)=O C(=O)(N1CCC(c2ccccc2)O1)c1cc(C)c(C)s1 N1(C(C(C#C)(C)C)=O)CCOC2(C1)CN(C(c1cnc(OC)s1)=O)C2 C1(CNC(COC2CCCC(C)C2)=O)N(C(=O)CCC2CC2)CCCC1(C)C c1(SCC(=O)NC(C(C)(C)NC(C2C(C#C)C2(C)C)=O)C)ccc(F)c(F)c1 N1(C(c2c(C)occ2)=O)Cc2nccn2CC(NC(C2Cc3nccn3C2)=O)C1 C#CC1(N(C)CCC(=O)OC)CCN(C(=O)C(=O)Nc2cccc(C)c2Br)CC1 c1(CNC(CC2(C=C)CN(C(=O)COCC=C)C2)=O)ccc2nc(O)[nH]c2c1 c1(CN2C(C(N3CCOCC3C)=O)CC(=C)C2)c(F)cc(C)cc1F C1(NC(C2CCN(C(C)=O)C2)=O)CN(C(=O)COCCF)CC1O C1(CC(=O)NC2(C(=O)NCCC3CCCOC3)CC(CO)C2)OCCCO1 c1(OC)nccc2c1CN(C1CC(CS(N)(=O)=O)C1)CC2 CC(C)(Cc1ccccc1)C(=O)OCc1ccccc1.c12cc(-c3cccs3)nn1C2 c1(C(N2CC(C)(NC(C3CC(CN(C)C)C3)=O)C2)=O)cccc(C2CCOC2)c1 c1(CC(=O)NCC(CC)NC(c2ccccc2OC(F)(F)F)=O)c(C)cnn1C C1(C)(C(=O)NC2(c3ccc(C(=O)OC)cc3)CCOCC2)C2CCCCC12 N1(C(c2c(CCNC(C3N(C)CCCCC3)=O)n[nH]c2)=O)CCOC2(CCC2)C1 c1(C(N(CCN(C(=O)Cn2cnnc2)CC)CC)=O)nn(C)cc1S(C)(=O)=O c1(C(=O)NCC(CC)NC(=O)C2=CC3CCCC23)cc(N)cc(S(C)(=O)=O)c1 c1(C(N2CCC(OCCNC(c3ccc(F)c(Cl)c3)=O)C2)=O)ncnc(O)c1F N1(C(C(C(C)C)n2cncn2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC1CF c1(-n2cc(SCC(=O)NCc3c(SC)cccc3F)nn2)cccc([N+](=O)[O-])c1 C(=O)(C(O)C(C)(C)C)N(C)CC1(NC(=O)CCc2nnc(C3CCCC3)o2)CC1 C1(NC(CC(C)OC)=O)COC2(CCN(C(c3occc3C)=O)CC2)C1 C(C(=O)N(C1CCN(C(c2nocc2-c2ccccc2)=O)C1)C)(C(C)C)OCC Cc1nn(C)c(C)c1OCC(=O)NCC1(F)CC(NC(=O)CSCC(C)C)C1 N1(C2C3CN(C(C4(CO)CCC4)=O)C(C3)C2)CCC(CO)C(F)(F)C1 Cc1cc(C(=O)NC(C(=O)NC2CC3(CC3)C2)c2ccoc2)ccn1 c1(C(CCC(=O)NCCCNC(=O)CC23CCC(CC2)C3)=O)cc(F)ccc1F N1(C(C(=O)NC2CCCCC2)C2CCCC2)C2CCC(O)C1CCC2O S(=O)(=O)(c1cc(Cl)ccc1Cl)N1C(C)(C(=O)NC2CCN(C(=O)C3CC3)C2)CC1 N1(Cc2sc(C(=O)OC)c(C)n2)CC2CC(NC(=O)CCCCCBr)CC2C1 c1(C(=O)NCc2ccc(NC(C3N(C(C)=O)CCC3)=O)cn2)cnc(O)c(C)c1 CC1COc2c(C(=O)NCC(CNC(c3cnc(Cl)cc3N)=O)CO)cccc21 c1(C(=O)NC(CC)C(=O)NC2CCC=CCCC2)cnn2ccccc12 CCCC(C)C(=O)N1CCOC(CNC(=O)CNc2cccc(F)n2)C1 c1(OC)cc(C(N2CCC3(NC(=O)CSC)CCCC23)=O)cc(Br)c1OC C1(C(=O)NCC2CCN(C(c3nc(OC)c(F)cn3)=O)C2)CCCCC(F)(F)C1 N1(C(CCCC(=O)NCC)=O)CC2=C(C1)CN(C(=O)C(C)(O)CC(C)C)C2 C1(C(=O)NCc2c(C)noc2C)CC(C)CN(C(=O)CSc2ccccn2)C1 c1(CC)ccc(-n2cc(C(=O)NC3CCC3NC(=O)CS(N)(=O)=O)nn2)cc1 C12(C(N(CC3(C)CNC(=O)O3)C)=O)CCCN(CCC1)C2.C(=O)(C(C)(C)C1CCCO1)N c1(C(=O)NC(CC(C)NC(c2c(CC)c(C)sc2)=O)C)cccc([N+](=O)[O-])c1 C(=O)(C1=CCCC1C)NC1CC(CCC(=O)NC(c2ccoc2)C)C1 C1(C(=O)NCC2(F)CC(NC(C(Cn3ccc(C)n3)C)=O)C2)COCC(C)(C)O1 C(=O)(C(O)CC[S+](C)C)N1C(CNC(CN(CCC#C)C)=O)CCC1 CP(C)(=O)C1CCCCC1C(=O)N(CCNC(=O)Cc1cncnc1)C1CC1 Cc1cnn(C)c1C(=O)NCC=CCC(=O)NC1CC(N(C)C(C)=O)C1(C)C c1(OC)ccc(C(=O)NC2CCC2NC(=O)CC2(C)CCCC2)c(Br)c1 N1(C(CC(CC)C(C)(C)C)=O)CCC2(CC1)CN(C(=O)CCC(N)=O)CC2CO c1(-c2n(-c3nccc(C)n3)ccn2)cc(C(=O)O)c(N)cc1F N1(C(C2C(C)(C)CCO2)=O)CCC(C(=O)NCC2(C)CCCS2)=C(F)C1 C1(CNC(=O)C=CCO)CCC2(CCC2)CN1C(C1COCCO1)=O CCC(C)C(C(=O)NCC1CC(NC(C2C3CCCC23)=O)C1)OC c1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)CC)cc2cccnc2[nH]1 C=CC(C)(C)CC(=O)NC1CC(OC)CN(C(=O)CN2CCCC2CO)C1 c1(C(=O)NCC(CN(C)C(c2c[nH]nc2C2CC2)=O)(C)C)cn(C)nc1O c1(OC)ccc2cc(C(=O)N(CC(O)CNC(c3cncn3C)=O)C)ccc2n1 N1(C(c2cc(COC)no2)=O)CC(NC(C2CCS2(=O)=O)=O)CCC1C C1(NC(C=CC2(C)COC2)=O)CCCCN(C(C2CC(O)C2)=O)C1 c1(C(=O)NCCCN(C(CCC#CC)=O)C(C)C)ncsc1S(N)(=O)=O C1(C(=O)NC(CO)C(C)NC(C2COCCO2)=O)(OC)CCOC1 Cc1cc(C(=O)NCC(CNC(=O)C(F)n2cccn2)CO)n(C)n1 N1(C(c2ncc(N)nc2)=O)CC2CCN(C(C3CCCC4(CC4)C3)=O)CC12 c1(OC)ncnc(C)c1NC(C12CC(CO1)N(C(=O)CN1C(=O)CNC1=O)C2)=O C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C12OCC(NC(CCCCCC=C)=O)(C1)C2 O=C(CCCCC(F)F)NCCC1CCCCN1C(c1cc2sccc2cn1)=O N1(C(CNS(CC)(=O)=O)=O)CCOCC1CC(N1CCCCC1C(F)F)=O CC1CCCN(n2nc(C3CCCCC3)nc2-c2ccc(C(F)(F)F)nc2)C1 C1(N(CC)CC)CC1N=c1[nH]c(N(C)C)nc2ncn(C)c12.c12csc(n1)CN2 C1(NC(CCSc2nc(C)[nH]n2)=O)CCN(C(=O)CC=C(Cl)Cl)CC12CCC2 N1(C(c2cn(C)nn2)=O)CC2CCCC(NC(=O)CSCC(N)=O)C2C1 N1(C(C(C)SCCCC)=O)CC(C2CCCCN(C(=O)COCC3CC3)C2)C1 Cn1ncc(C(=O)NOCC(=O)N(c2ccc(F)cc2)C2CC2)c1N CC1(CNC(C2CCC(F)C2)=O)CC(F)(F)CN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(C(N(CCNC(C2CCC(C)S2)=O)C2CC2)=O)ccc(N)c2c1CCCC2 CCCCC(O)C(=O)N1CCC(CNCc2ccc(C#N)cc2)CC1 c1(C(=O)NC(C(=O)N(CCC2CC2)CC)CO)ccc(C#N)[nH]1 C1(c2nnnn2CC(F)F)(NCCC(=O)NC)CN(C)CC1C N1(C(C(C)NC(CC)(C)C)=O)CC(NC(C2(C)CC2Br)=O)CC2(CC2)C1 C(=O)(CC(C)CC(C)(C)C)N1CC(C)N(C(c2ccc(=O)n(CC(C)O)c2)=O)CC1 C1(C(=O)NC(C2CCN(C(CC(C)(F)F)=O)CC2)(C)C)CCC12CCOCC2 CN1CCN(C2CCN(CC(=O)Nc3ccccc3Cl)CC2)C1=O c1(CN(C(=O)NCC2C3CN(CC(F)(F)F)CC23)C2CC2)cc(F)c(F)cc1F CC(=O)CCCC(=O)N1CC(F)CC1C(N1CCC(CCN(C)C)CC1)=O c1(C(=O)NCc2cccc(CNC(CSCC)=O)c2)cccc(C#N)c1C C(C(C)(C)C(=O)NCC(C)(CO)NC(c1coc(C(F)F)c1)=O)SC C(=O)(CCN1C(=O)NCc2ccccc21)NC(c1c(C)n(C)nc1)C N1(C(CCc2cc(C)[nH]n2)=O)CCC(NC(=O)CN2CC(C)(C)C2)C1(C)C N1(C(c2cccc(OC)c2N)=O)CCCCC(C2CN(C(=O)C3=CCC3)C2)C1 N1(C(C2CC(OCC)C2)=O)CC=C(CNC(=O)CCc2nc(C)no2)CC1 c1(OC)ccc(C)c(C(=O)NCC2C=CCN2C(c2cccc(N(C)C)n2)=O)c1 c1(C(=O)NC2CCN(C(C3(C)CC3(F)F)=O)CC2F)ccc2ncccn12 C(=O)(CCCCC#N)NCCCc1cc(C(=O)NCc2n(C)nnn2)no1 c1(N2CCC(F)(F)C2)nc2c(c(=NC3COc4cccc(F)c4C3)[nH]1)CSC2 N1(C(CC2(C#N)CCC2)=O)CC2CC2(CNC(c2ccnc(C(F)(F)F)c2)=O)C1 CN1CC2(CCCN(CCN3C(=O)NC(C)(c4ccc(Br)cc4)C3=O)C2)CC1=O c1(C(=O)NC2(C)CCCN(C(=O)COC3CCC3)C2)cccc2c1OCCN2 C1(CNC(=O)NC(c2c(C)scn2)C)CCC2(CCC2)O1 C1(COC)CN(C(C2(SC)CCC2)=O)CCN1C(=O)C(F)OC Cc1ccc(F)c(N2CCCC(NC(=O)C(C(C)C)n3cnc(C)c3)C2=O)c1 N1(C(c2ncc(C)nc2)=O)CCC(CNC(=O)C(C)Cc2cnco2)C(C)C1 C=CC(C)(CC)C(=O)NCC(CO)NC(=O)CCCOc1ccc(F)cc1 N1(C(C(C)(C)NC(C2CC(=C)C2)=O)=O)CCC(O)(CO)CC1 Cc1nnc(CNC(N2CCC2c2ccccc2)=O)o1.c12ccn(n1)C2 C1(CNC(CSSC)=O)CCCC12CC2.C12(CCC1)C(=O)NCC2 N1(CC(=O)NCC2(NC(C3N(CC)CCC3)=O)CCOC2)C(=O)NC(C)(C)C1=O c1(C(=O)NC2(CCCNC(CC(C=C)C)=O)CC2)ccc(OC)nc1Cl C(C(=O)NC(C)CC1COC1)(C(C)(C)C)NC(CCOCCOCC)=O C1(CNC(c2ncccc2O)=O)CCC2CN(C(C3(CC4CCC4)CC3)=O)CC12 C(=O)(C(F)(F)CCn1cccn1)N(CCNc1nccc(C)c1O)CC Nc1c(F)ccc(Cl)c1C(=O)NCCCOCCNC(=O)C1=C(Cl)CCCC1 CC(C)CC(C(=O)NC12CC(C1)N(C(C1(C)CCC(O)CC1)=O)C2)n1ccnc1 C(=O)(C(C)(C)CC(F)F)NCC(CCCC)NC(c1cncc2n[nH]cc12)=O O=C(N=c1nc2cc(Cl)ccn2[nH]1)N(c1ccc([N+](=O)[O-])cc1)C c1(OC(C)C)ccc(C(N2CCC(N(C(=O)CCOC3CCC3)C)C2)=O)c(F)c1 Cc1cc(C)c(C(=O)N(C2CN(C(c3ccncc3Cl)=O)C2)C)[nH]1 CCCCC(CC)C(=O)NCC1CN(C(c2cnc(O)n2C)=O)C1 C1(CNC(=NCCC=C)NC2CC2C)COc2cc(OC)ccc2C1 N1(C(c2c(C)occ2C(F)(F)F)=O)CCC(C2CCN(C(=O)C3CC3)C2)CC1 c1(C(C#C)OC(C)CC)ccccc1 c1(SC)nn(CNC(NCCC(C)(C)OC)=S)cc1Br c1(C(=O)NCC=C)nc(C(=O)NC2CC(NC(=O)C(C#N)C3CC3)C2)cs1 C1(C)(NC(C2(F)CCN(C(CC3CCN(C)CC3)=O)C2)=O)CCCC(C)(C)C1 c1(C(N2CC(CC(C)NC(=O)CC3CCC(=O)NC3)C2)=O)cccnc1S c1(N(CCC(=O)NO)C(C2CC3CCC3C2)=O)ccccc1Cl C12(CC)CCC(C(=O)N(C3CCN(C(C4CC5CCC4C5)=O)C3)C)(CC1)CO2 c1(C(N(C)CC2C3CN(C(CC(=O)NCC)=O)CC32)=O)cccc(OC)c1F c1(C(N(C)CC2(CNC(c3cc4sccc4s3)=O)CC2)=O)cncn(C)c1=O O(C1CCc2c(F)cccc21)C(c1cc(F)cc2c1CCC2)=O N1(C(c2c(OC)cc(F)cc2)=O)CCC(C(=O)NC2(C(N)=O)CC2)C(C)(C)C1 c1(C(N2C(CNC(C3CCCO3)=O)CC(OC)C2)=O)cc2c(C)ccc(F)c2[nH]1 CCC(C)CCCCC(=O)NC1C=CC(C2CCCN2CCOCC2CC2)C1 c12ccc(cc1)N(CCOC)CCNC2=O.C(=O)(C(F)=CCCF)NCCN(C)C c1(C(=O)NCC2N(C(C(CC=CCC)C)=O)CC2)ccc(C)c(NS(C)(=O)=O)c1 CC1C(C(=O)NCC(=O)N(C)O)CCN1C(=O)CCCCC1CC1 c1(OC(C)C)cnc(C(=O)NC2CCOC2C)cn1 c1(C(=O)NCC(C)(CO)NC(C2CCCS2)=O)nc2c(s1)COCC2 c1(C(=O)NCCCCN(C(=O)N2CCCO2)CC)ccc(OC)c(F)c1 N1(C(c2c(C)cncc2C)=O)CCC2CC1CN(C(=O)CN(C)C)C2.O1NN(C)C1 c1(C(N(C2CCC(NC(=O)C(=Cc3cscn3)F)C2)C)=O)cc2n(n1)CCCN2 c1(C(=O)NC2(C(=O)NC(CCOC)COC)CCC2)cccc(C)c1C c1(C(N2CCC3CN(S(=O)(=O)c4ccncc4)CC23)=O)ccc(Br)c(F)c1F C(N=c1cc(C2CC2)nc(Cl)[nH]1)C1(CNC(C2C(OC)CCCC2)=O)CCC1 n1(CCC)ccc(NC(C2(CC)CN(Cc3cnc(Cl)s3)C2)=O)n1 C(=O)(C(C)C(C)NC(=O)C=C(C)CNC(c1cc(Cl)n(C)n1)=O)OC c1(OC)cccc(OC)c1NC(c1cnc(C2CCOCC2)nc1C)=O c1(C(=O)NC2(CNC(CC(CCC)O)=O)CCCC2)cc2cnccc2o1 N1(C(C2CCC(=C)CC2)=O)CCC2(CCCN(C(=O)CC(F)(F)C(F)(F)F)C2)C1 N1(C(c2ccc(C#C)nc2)=O)CCN(C(=O)CCc2cn(C)nn2)CC(O)C1 c1(OC)cccnc1C(=O)NCC(C)(C)CNC(c1cn(CCF)nn1)=O CC1CN(C(=O)CCCN=[N+]=[N-])CC2(CCN(C(c3ccnn(C)c3=O)=O)CC2)O1 Cc1cc(NC(C2(C)CCCN2Cc2ccc(F)nc2)=O)ccc1C#N CC1CCCN(C(=O)Cc2cccc(OC(F)F)c2)C1CNC(=O)COCCF c1(CNC(C(CN(C)C)NC(=O)COC2CCOC2)=O)ccc(F)cc1F N1(C(C)C)CC(C(N2CCC(N(C)C(c3cn(CC(N)=O)nn3)=O)C2)=O)CC1=O c1(C(=O)NCCNC(CC2(C)CC2(F)F)=O)ccc(N)cc1C(F)(F)F C(C)(CCCCNC(c1ccc(F)cn1)=O)NC(CC(=C)Br)=O C1(CNC(CC=C=C)=O)C(O)C(O)CN1C(c1cc(CF)on1)=O CN1CCn2cc(C(=O)NCCCCNC(=O)CN(C3CCCC3)C)nc2C1=O C(CCCC(=O)NC(c1ccc(C(C)(F)F)cn1)C)OCCOC Nc1cc(Cl)nc(Cl)c1C(=O)NCC1CCC(NC(C2CCCC23CCC3)=O)C1 C1(C(=O)NCC(CO)NC(c2c(C(C)C)noc2)=O)CCc2nccn2C1 Cc1cc(C(=O)NCC2COCCN2C(c2scc(Br)c2Br)=O)cc(Br)c1 Cc1cc(C#N)ccc1NC(=O)COCP(C)(C)=O.N12CCN(CC1)CC2=O C1(Nc2ccc(N(C)C)cc2)CCC2(C1)CN(C(c1ccc(Cl)cc1)=O)C2 C1(O)(CNC(C2CC(N(C)C)C2)=O)CCCN(C(c2ccc(Cl)c(N)c2)=O)CC1 c1(C(N2CC(O)(CNC(c3ccnc(C(F)(F)F)n3)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(c2cc(CC)n(C)n2)=O)CC2CCC(NC(=O)Cc3cncn3C)CC2C1 C(=O)(CC(C)(C)N1CCOCC1)NC(CCNC(C1C(COC)C1)=O)C Cc1cncc(C(=O)NC2CCC(F)(CNC(c3nc(Cl)c(Cl)s3)=O)C2)n1 N1(C(COCC(C)C)=O)CCCN(C(c2ccc(F)cc2C(F)(F)F)=O)CC1 C=CCC(CC(C)C)C(=O)NCC(C)(C)CN(C)C(c1ccc(C(C)C)cn1)=O c1(C(=O)NC(C(=O)NCCC(CC)O)Cn2cccn2)ccc(C)c(C)c1 c1(CCC(=O)NCC=CCNC(C2CCC(C)CC2)=O)cc2ccccc2o1 n1(CCOC)ccc(=NC(=O)CNC(=O)N=c2[nH]nc(C(C)(C)C)s2)[nH]1 N1(CC)CC2CN(C(C3CN(C(=O)C=CCOC)CC(C)(C)C3)=O)CC2C1 CC(C)(C(=O)N1CC(C(F)(F)F)C(CNC(c2ccns2)=O)C1)S(=O)(=O)C1CC1 C1(NC(c2c[nH]nc2C2CC2)=O)CCC(NC(C2(C(F)(F)F)CC2)=O)CC1.C1(S)CC1 N#CC1CCN(C(C2CC23CCN(Cc2ccc(-c4cc[nH]n4)cc2)C3)=O)CC1 N1(C(C=CC)=O)CCN(CCCCCC2CCCN(C(=O)C(=O)N(C)C)C2)CC1 C1(CC(=O)N(C)CC2(F)CCC2)CCN(C(=O)Cn2cnnc2O)C1 CCC(CCC(=O)NCCC(C)N(C(=O)C(c1ccc(C)o1)C)C)OC C1(C)(C(N(CCc2ccc(C)s2)C)=O)CC12CCN(CC(=O)NC(C)C)CC2 c1(C(N2CCCCC2CC(N)=O)C(=O)NC(C(=O)NC)C)ccc([N+](=O)[O-])cc1 CC1=C(C(=O)NC2CC3CN(C(=O)C=Cc4ccncc4)CC23)CCO1 C#Cc1cccc(C(=O)NC2CC(C)N(C(C3CCC4C(C3)C4(F)F)=O)C2)c1F c1(-c2nc(C(C)C)nn2-c2ccc(OC(F)(F)F)cc2)cn2ccccc2n1 C1(NC(C=CCNC(C(C)NC=O)=O)=O)CC12CCCC2 C(=O)(C1=Cc2cc(F)ccc2OC1)N1CCC(Nc2ccnc(C)n2)C1 N1(C(CC(CNC(c2cn(CCC)nn2)=O)C)=O)CC(F)(F)CC1C(=O)NC C1(c2noc(-c3ccc(OCC(C)C)o3)n2)(NC(C(CC)SC)=O)CCCCC1 N1(C(C(CC2CC2)NC(c2cc(Cl)no2)=O)=O)CCCC2(C1)N=N2 C(CCC(=O)NCC1(C(=O)NC(CSC)CC)CCCC1)=CC CN1C(=O)CCC1CNC(CC(=O)NCc1ccc(Cl)o1)CC1CC1 N1(C(C2C(CCC)CCC2)=O)CCC2CCCC12CNC(C1(N(C)C)CC1)=O C1(CCNC(=O)C=NOC)(NC(C(CC)C)=O)CCOCC1 N1(C(C23N(C(C(C(CC)C)N(C)C)=O)CC(C2)C3)=O)CCOC2COCC12 C1(C(=O)NCC2C(OCC)CC2)C2CC(O)C(C2)N1C(=O)C1=CCCCC1 N1(CC(=O)NCC(CN(C(C2C(C(=O)NCC#C)C2)=O)CC)C)CCCNS1(=O)=O C(=O)(CC(=O)N(CC(C)NC(c1cc(CS(C)(=O)=O)on1)=O)CC)NCC c1(N2CCC(C3(C)CC3)C2)nc2ccc(Cl)cc2c(=NCC2(C)CCCCC2)[nH]1 CS(=O)(=O)c1ccc(C(NC=CC(=O)C(F)(F)F)=O)cc1Br.C12CC1C(=O)N2 c1(C(=O)NCCC(=O)N(C(C)COC)CC)cn(CC2CC2)nn1 Clc1ccc2c(CNC3(c4nn[nH]n4)CC34CCOCC4)c[nH]c2c1 c1(C(C(=O)NCC(CCOC)NC(=O)CCC2CCC2)C)ccc(OCC)cc1 N1(C(c2nccn2CCC)C(=O)NCC(=C)C)CCOC(C)(CC)C1 CC(C)(C)CC(=O)NCC1(F)CCN(C(C2CC(N3CCCC3)C2)=O)C1 N1(C(CN(C(C)C)C)=O)CC2CCC(C1)C2NC(C1CCCC(=O)N1)=O C12CCOCC1C(=O)N2.C1(CCOC)(NC(c2c(CC)cco2)=O)CCCC1 c1(CC)cccc(C(N2CCN(C(=O)C(n3nc(C)cc3C)C)CC2)=O)c1N CC(C)(C)[Si](C)(C)OCCNCCCOC1(CCOCCc2ccccc2)CCC1 C1(NC(c2c(C)n[nH]c2)=O)CCC(CNC(=O)C(O)c2ccsc2)CC1 c1(OCCCC)ccc(CCN(C2CCN(C(=O)C(C)CC)CC2)C)cc1 c1(C(=O)NC2CC(O)(CNC(C3(OCC)CCC3)=O)C2)cc(C)c(C)cn1 c1(CCCC(=O)NCCCCN2CCCOC2=O)ccc(Cl)cc1 N1(C(c2cc(CCNC(C(NOC)=O)=O)on2)=O)C2C=CCC1CC2 C(C)(C)(CC(=O)NCC(N)=O)N(C(=O)Cc1ccon1)C N(C1CCCc2c1cnn2C)C(c1c(OC)c(F)ccc1)=O N1(C(=O)CCCc2cccs2)CCC2(CCCN(C(=O)CCc3cnn[nH]3)C2)C1 Cc1cnc(F)cc1-c1ccc(NC(C2CCCN2C(=O)CNC(C)C)=O)s1 C12(CNC(CCc3c[nH]c(=N)[nH]3)=O)CCC1CN(C(c1ccc(Cl)cc1Cl)=O)C2 c1(-c2ccc(CC(=O)NC(=O)NCCCOC)cc2)ccc(C(C)C)c(F)c1 CCCCC(C)CCC(=O)N1CCCC(NC(c2cc(C)cc(C)c2C)=O)CC1 C1(C)(OC)CCN(C(c2ccc(-c3cn(C)nc3C)cc2)=O)C1 C#CCC(C(=O)Nn1cnnc1C)NC(=O)C1=CCOCC1 c1(C(N2C(CNC(C(CCC)CC)=O)C=CC2)=O)cnc(C)c(Cl)c1Br C1(CC(=O)OC)CCN(C(=O)C(C2CCN(C(=O)CSC)C2)F)CC1 Cc1c[nH]nc1C(=O)NC(C)CC(=O)NCCCN(C)C(C)C C(=O)(C(C)(C)C(C)(C)C)N1CC(c2cn(C(C(=O)N(CCSC)CC)C)nn2)(F)C1 C(=O)(C(C)C(C)c1ccccc1Cl)NCC(C)N(C(CC)(C)C)C C1(N(C(c2ccc(C(C)C)o2)=O)C)CN(C(c2coc(Cl)n2)=O)CC12CC2 C1(NC(c2c(C(C)C)con2)=O)CCC2(CC1)CN(C(=O)CN(C)CCOC)C2 c1(C(N2CCN(C(C3CC(SC)C3)=O)C3(C2)CC3)=O)cc2c(C)cccn2n1 c1(C(C(=O)NC(C)C2CC2)N(CCCC#C)C)nocc1C(C)C CC(C)(CS(C)(=O)=O)C(=O)N1CC2CC(C1)N(C(=O)Cc1cccnc1O)C2 C(=O)(C1CCCn2cc(C(F)(F)F)nc21)N1CC(NC(CCCC(C)(F)F)=O)C1 N1(C(C2CCC(C(=O)O)C2)=O)CCC(O)(Cc2cn(CC3CCC3)nn2)CC1 c1(NC(C2(NC(C3C=C(C)CS3)=O)CC(O)C2)=O)ccc(Cl)cc1C c1(NC)snc(C)c1C(N1CC2CC2(NC(=O)CC2(C(F)(F)F)CC2)C1)=O N1(C(c2c(CC(=O)OC)occ2)=O)CC2(CCCC2NC(=O)CCCC(C)O)C1 Cc1cc(C)c(NC(C2(C)CCCN(C(c3ccc(Br)c(Cl)c3)=O)C2)=O)cn1 C=C(C)CCC(=O)N(C1CCCCC1NC(=O)Cc1nc(C)sc1Cl)C C(=O)(CC(C)(C)C1CC1)N(C(C)CCNC(C1CCCN1C1CCOCC1)=O)C C1(NC(Cc2n(C)cnc2)=O)(CNC(=O)CC#N)CCCCCC1 C1(CNC(c2ccc(O)nc2)=O)CC2CCC1N2C(=O)CCC1CCC1 C1(C(C)NC(=O)CCn2cncn2)CCN(C(c2nc[nH]c2C(F)(F)F)=O)CC1 C1(NC(CC=CC)=O)CCN(C(c2cnnc3ccsc23)=O)CCC1CO C(=O)(C1Cc2ccc(Cl)cc21)NCCCCCCNC(C(C(=O)OCC)F)=O N1(C(CS(=O)(=O)NC)=O)CCN(C(c2cccc(CO)n2)=O)C(C)C1 c1(C(=O)NC(C)(C)CCNC(C2CC2Cl)=O)cc2c(cc1N)OCO2 N1(C(COCCCC)=O)CCC(NC(=O)Cc2ncc(C)[nH]2)C(O)C1 C12(CNC(c3cnc(CCC)s3)=O)CC1CN(C(=O)C(CC)c1ccccc1)C2 c1(C(N(C2CN(C(Cc3nc(COC)sc3)=O)C2)C)=O)cccc2nc(C)nn12 C1(CC(=O)NCCSCC(=O)NCc2ccnn2C2CC2)CC2CC2C1 C1(COC(C(C)CC2CCCCO2)=O)CC2c3ccccc3CCC12 CCCC(C(O)C(=O)NCC1CCCC1)NC(=O)C(c1cncn1C)O C1(NC(C=COCC)=O)CCN(C(c2ccc(OC)c(Cl)c2)=O)CC1F c1(CC)ccccc1-n1cc(CNC(Cc2ccccc2)CCO)nn1 C1(C(=O)NCc2c(N3CCC(C)CC3)cccc2)CC(O)C12CCC2 C(=O)(C1=NN(CCO)C(=O)CC1)NC1CCCC(NC(C(C)N(C)C)=O)C1 c1(C(C)=O)ccc(C(N2CCCC(c3cn[nH]c3)C2)=O)cc1F C1(C)(C(=O)NC2CCCN(C(C)=O)C2)CN(C(=O)C(C)n2cncn2)C(C)(C)C1 C(=O)(NN1CC(C)N(C)C1=O)c1c(C)sc(C)c1C C(C)(C(CC(=O)NCCC(O)CO)NC(=O)CC1CC(C)=NO1)OC C(=O)(C1=NOC2COCC12)NC1CCC(CNC(c2[nH]nc(C(C)(C)C)n2)=O)CC1 c1(NC(C2CCC(NC(=O)NC(C3(CC)CCC3)C)C2)=O)ccc(CC#N)cc1 n1(CC)cc(C(=O)NC(C)(C)CN(C(=O)CCCCOC)C)c(C)n1 CC(C)C(CCNC(=O)CSCC(N)=O)NC(c1csc(-c2ccccc2)c1)=O c1(C(N2CCC(C)(CNC(CCC#C)=O)C2)=O)sc2cccc(F)c2c1COC C1(C(=O)NCC(CC=C)NC(c2cc(C(F)(F)F)nn2C)=O)CC2CCC1C2 N1(C(CON2CC(C)(C)OC2=O)=O)CCOc2cccc(F)c2C1 N1(C(C2(C)C(C)CCC2)=O)CCC2(CCN(C(c3cc(C(F)F)no3)=O)C2)C1 N1(CCCC(=O)NC2CC(O)C2)C(=O)CCC1=O C(=O)(C1=C(F)CN(C(C2CCCCNC2=O)=O)CC1)N1CC(C)C(N(C)C)C1 c1(C(C)C)nc(NCCC(C)(C)C)cc(=NCC(C)(Cc2ccccc2)CO)[nH]1 C1(NC(C(c2ccc(C(F)(F)F)cc2)N(CC(C)C)CCC)=O)CCCCCC1 CC1(C(=O)NC2CCC(NC(=O)Cn3cc(Cl)cn3)CC2)COC(=O)C1 n1(CC)nnc2cc(C(=O)NC(C)CNC(C3CCCC3C)=O)ccc12 S(=O)(=O)(c1cc2c(cc1Cl)OCCCO2)N1C(CC)COC(C)C1 N1(C(C2CC(C(=O)OC)C2)=O)CCCC2(CCCN2C(c2cc(N)c(Cl)cn2)=O)C1 C(CN=c1[nH]c2c(c(=NCC3(C)CC3(C)C)[nH]1)SCC2)c1n(C)ncn1 c1(C(=O)NC(CNC(C2(C)CCN(C(C)=O)C2)=O)(C)C)c[nH]c2cccnc12 N=c1[nH]cncc1C(N1CCOC(C(N2CC(NC(N)=O)C2)=O)C1)=O C1(C(N2CC(CN(C(Cc3nc(C)c(C)[nH]3)=O)C)OCC2)=O)CC(C)(C)CCO1 Cc1ccc(F)c(NC(=O)C(CNC(=O)Cc2c[nH]nc2C)CC2CC2)c1 c1(NC2(CNC(Cc3c(C)cccn3)=O)CCC2)cc(C)c([N+](=O)[O-])c(C#N)c1 c1(OC(CNC(NCC(C)OC)=S)(C)C)ccc2c(c1)CCCC2 N1(C(C(CC=CC)CC)=O)CCC2CCCC12C(=O)NCCN(C)C C(CC(C)(C)C(F)(F)F)NC(c1n(C)nnn1)c1c[nH]nc1-c1ccc(Cl)cn1 C1(NC(c2ccc(CC)cn2)=O)(CNC(=O)Cc2c[nH]nc2C)CCCCCC1 C(=O)(CC(C)C(F)F)N1CC(Cn2cc(NC(=O)NC3CCCC(CC)C3)nn2)C1 N1(C(C(C)OCC2(CCN(C)C)CC2)=O)CCC(C)(C(=O)NC(N)=O)C1 Cc1cnc(N(C(C)CCNC(=O)NC2CC2CC(C)C)C)o1 C1(CNC(C2(C(=O)NCC)CC2)=O)CN(CC2CCCC2)CCO1 C=CC(C)(CCOC)C(=O)N1CCN(C(=O)C(F)=CCC)C(CCO)C1 N12CCC(F)(F)C(C1)C(=O)OCC(=O)NCCS2(=O)=O.CCOCC N1(C(C(CC)C)=O)CC(OC)CC1C(=O)NCC1CCCC1N(C)C N1(C(C(c2ccc(N)cc2)C)=O)CCC(C(C)NC(C2CC=CC2)=O)CC1 C1(OC)(CNC(C2CCC2)=O)CCN(C(=O)C(C)(O)C2CC2)C1 C1(CNC(CSCC(C)=O)=O)C2CN(C(C3(C)CC3c3ccccc3)=O)CC12 c1(NC(=O)Cc2cn(C3(NC(C4CCC(F)C4)=O)CC3)cn2)ccc(O)c(Cl)c1 C1(c2n(CCCOC)nnn2)(NCc2cc(OC)ccc2C)CCCN(C)CC1 c1(OC)cc(CN2CCC2(C)C(=O)Nc2cc(C)cnc2Br)c([N+](=O)[O-])cc1O C1(C(=O)OCC)C2CCC1(C(=O)NC1CCCC1NC(=O)C(C(C)O)N(C)C)C2 C(=O)(C(C1=NOC2CC12)N1CCc2nc(Br)sc2C1)NCCCCCC CCC(C)(CO)C(=O)N1CCC(C)(CNC(C2(c3cccc(OC)n3)CC2)=O)C1 n1(C(C)(C)C)nnnc1C(C1(C2CCCC2)CC1)NC(C1CCCCC1)NC1CC1 O=C(C1OCCc2ccccc21)NC1CC(O)CN(C(C2CCSCC2)=O)C1 c1(CC(=O)NC(C(C)C)CCNC(=O)C(c2nccn2C)C)cccc(Cl)c1Cl c1(N(CC(C2CC2)OC)C)nc(=NCCC(C)(C)C)[nH]c2ncn(C)c12 c1(C(N(C(C)C(=O)NCCc2cc(C)ns2)CCC)=O)ccc(C)cc1F C(CCCC(=O)N(C1CC1)C1CC1)N(CC(C)CCO)C CCCC(C#N)C(=O)N1CCC(C(=O)NC2CC(CO)(CO)C2)C1(C)C C1(N(C(C(C)NC(N)=O)=O)C)CCCN(Cc2ccc(CN)s2)CC1 C(=O)(C#CC1CCOCC1)NCC1(C2(O)CN(C(C(CCCCC)F)=O)C2)CC1 N#CC1CCN(C(c2cncc(NCc3cc(Br)co3)c2)=O)C1 CC1CCCN(C(C2CCCN(C(C3CCOC3)=O)C2)=O)C1CO Cc1oc(C(C)C)cc1C(=O)NC1CC(C)(NC(=O)CCCn2cccn2)C1 Cc1cc(F)c(C(N2CC(NC(c3cc(O)nc(Cl)c3)=O)C(F)C2)=O)cc1F c1(C(=O)NC2C(C(=O)Nc3n(CC)ncc3)CCC2)ccc2nccn2n1 C1(CC)CN(C(=O)COC)CCC1NC(c1c(C)cnn1C)=O N1(C(CC(C)C)C(=O)N2CC(C(C)(F)F)C2)CCc2ccccc2C1 CC12CC(C1)C(C(N1CCC(NC(=O)COc3ccc(F)nc3)CC1)=O)CO2 c1(CN2CCC(N(C)C)C2)c(Cl)cccc1I.c12sccc1NC2=O C1(F)(CNC(c2cc(C)sc2)=O)CCCN(C(=O)Cc2ccc(Cl)cc2Br)C1 Cc1c(C(N2CCC3CN(C(=O)C=CC(=O)N(C)C)CC23)=O)sc2cc(F)ccc12 CCCCC(C(=O)NCCOCC(N1CCOC2CCC12)=O)OC n1(CC(=O)NCC2(F)CN(C(C3=C(C)OCCC3)=O)C2)ccc2ccc(Cl)cc12 c1(OC)cc(Cl)cc(Cl)c1CO.N12CCC(C)(C(O)C1)C(=O)N1CCC(C1)C2=O c1(C(=O)NC(C)CNC(c2ccn(C)c2)=O)cc2cc(F)c(F)cc2[nH]1 CC1CC(CNC(c2cccnc2OCCO)=O)CN1C(=O)CCCNC(N)=O C1(NC(c2cnc(C)n2C)=O)C(C)CN(C(C2(c3cc[nH]n3)CC2)=O)CC1C C=CC1CN(C(c2c(C)nn(CCO)c2C)=O)CC1NC(=O)CCCNC(N)=O c1(-n2cc(C3(C)CCN(C(c4cc(N)ccc4Cl)=O)C3)nn2)cccc(Cl)c1Cl n1(C(C)C)cc(C(=O)NCC(C2CC2)NC(C2CC(=O)C2C(C)(C)C)=O)cn1 C1(C(N(CCCCCCNC(C(CCC)C)=O)C)=O)CC2CCCCC12 C1(CC(N2CCN(CCNC(C3(C)CC3(F)F)=O)CC2)=O)CCCC2(CCC2)O1 N1(C(c2cccc(C)c2)=O)CC(NC(C2(n3cccc3)CCCC2)=O)CC(O)C1 C(N=c1[nH]c(=NCCS(C)=O)[nH]c2c1CSC2)c1c(N(C)C)cccc1 c1(C(=O)NC2CN(C(CCOCC)=O)CC2N=[N+]=[N-])c[nH]c2cccnc12 c1(OC)ccc(C)nc1C(=O)NC(C)(C)CNC(=O)C(C)Cc1cccc(Cl)c1 CC1(CNC(C2CC3C=CC2O3)=O)CN(C(=O)CC2(O)CCOCC2)CCO1 CCC(C(=O)NC(C)CNC(c1ccn(-c2ccccc2F)n1)=O)C(C)(C)CC CC1(C(N2CCCC(C)(NC(C3CC4(CC4)C3)=O)C2)=O)CCC(F)(F)C1 c1(C(N2C(CNC(=O)Cc3cnoc3)CCC2)=O)coc2c1CSC2 CC1C(NC(=O)CC(O)C2CCCC2)CCN1C(=O)CSc1ccccc1Cl c1(C(N2CC(C(=O)NCCN)OCC2)=O)ccccc1[N+](=O)[O-] C1(C(=O)NCCNC(C(n2ccc(C3CC3)n2)C)=O)C2COCC12 c1(CCC)ncc(NC(=O)CN(C(C2SCC=C2C)=O)C2CC2)cn1 C(CNC(c1cn(C)nn1)=O)(CC(F)(F)F)NC(CCN(CC)CC)=O C1(C(=O)NCC(C)(CO)NC(C(C)C#N)=O)CN2CCN1CC2C CC(C)(C(=O)NCC1(NC(=O)CCCN2CCCCC2)CC1)c1cnc[nH]1 N1(C(C2CCN(C)C2)=O)CC2CC2C1CNC(C1(S(N)(=O)=O)CC1)=O C=CC(C)(O)C(=O)NCC1CC(C)N(C(=O)C=Cc2cncn2C)C1 N1(C2(C(=O)NCC(CC)NC(C3CCCC(=O)O3)=O)CC2)CCN(CC)CC1 C(=O)(C(C)(C)c1cnn(C)c1)NCCN(CCC)CC1COCCO1 Cc1ncc2ccc(C(N3CCC(O)C(NC(C4CC=CCC4)=O)C3)=O)cn12 Cc1nnc(NC(C2CN(C(c3ccnc(Cl)c3)=O)CCO2)C)c(C#N)c1C N1(C(c2n(COC)ncc2)=O)CC(CCNC(C2(CO)CCCC2)=O)OC(C)C1 c1(OCCCCC)cc(NCc2cncc(CC)c2)ccc1C CC1Cc2c(C(=O)O)cccc2C1NC(C1(n2cc(Br)cn2)CC1)=O c1(C(=O)NC(CNC(c2n(CC)nnc2)=O)CO)cc(S(C)(=O)=O)cc(C)c1F n1(CCC(N2C(CNC(C3(N(C)C)CCCC3)=O)CC2)=O)cnccc1=O N1(C(C)C)CC(C(=O)CCNC(c2cccc(Br)c2)CO)CC1=O C(c1cccn1C)=CC(=O)NC1CC(CNC(CC2N(C(C)C)CCC2)=O)C1 C(C1=CCN(C(c2ccn(C)c2-c2ccc(F)cc2)=O)CC1)NC(CC=C)=O c1(C(N2CC3(N(C(CC(C=C)C)=O)CC3)C2)=O)ccc2cc(Cl)ccc2n1 c1(C(=O)NC(CC)(C)CNC(c2cnnc(O)c2)=O)cc(O)nc(O)n1 c1(C(=O)NCC2(O)CN(C(c3c(C)ccc(OC)c3)=O)C2)ccc(O)c(F)c1F S(=O)(=O)(c1cc2cc(Br)cnc2o1)NCC1CCC(CC(=O)OC)CC1 C1(C(=O)NC2CC(NC(c3c(C)cc(F)c(N)c3)=O)C2)Cc2ccccc2C1C C1(CNC(C2N(C(c3c(C)nc(C(C)C)s3)=O)CC2)=O)CCC(C)(O)CC1 C1(NC(CCC2C(C)(C)C2)=O)CC(O)CN(C(=O)CCc2ccc(F)cc2Cl)C1 C12(C(N3CC(C4N(C(c5nnn(CC)c5C)=O)CCC4)C3)=O)CCC(CC1F)C2 c1(C(=O)NC2(CCNC(C=CC)=O)CCCC2)ccc2nccn2n1 C(=O)(C(CNC(C1(C2(C)CC2)CC1)=O)C(C)C)NC(C(=O)OC)CC1CC1 N1(C(C2CN(C(N)=O)C2)=O)CCOCC1CC(=O)NCc1nc(C2CC2)no1 Cc1ccc(Br)c(NC(CC2CCCN(CCN3CCCC3)C2)=O)c1F.C1C(=O)N1 C(=O)(C(C)(C)CC(F)F)NCC12N(C(Cc3cccc(C)c3)=O)CCC1CC2 Cc1ncc(C(=O)N(CCCC(N2CC3CC(C)C3C2)=O)CCCO)c(C)n1 c1(C(=O)NCCOCCN(C(c2cc(COC)sc2)=O)C)cccc2cncn12 Cc1nc2c(C(N3CCC(NC(C4CCC5CCCCN45)=O)C3)=O)cccc2o1 CN=c1[nH]c(=NCCN2CCC3CC23)[nH]c(=NCCCCC(N)=O)[nH]1 N#Cc1cncc(C(=O)NC2(C(=O)NCC3CC4(CCC4)CO3)CSC2)c1 C1(C(=O)NCC2CC2C#N)(CNC(COC2(C)CCC2)=O)CC2(CC2)C1 c1(C(=O)NCCC(C)NC(C=Cc2c(C)coc2C)=O)cccc2nccn12 CCCCC(F)C(=O)N1CC2CC(C(=O)NCCc3[nH]cnc3C)(C2)C1 Cc1[nH]c(=N)sc1C(N1CCC(CN(C)C(C2CCCC2)=O)C1)=O N1(C(CCC(C)NC(C2(NC(N)=O)CC2)=O)=O)CCC2CCN(C)CC12 c1(CCC(=O)NC(CC=C)CNC(C2CC(OC)C2)=O)ccc(Cl)c(OC)c1 c1(OC)cc(C(N2CCN(C(c3cnn(C(C)C)c3)=O)C(CF)C2)=O)ccc1O c1(C(=O)NC2(C)CCN(C(c3c(C)onc3C3CC3)=O)C2)cc(F)c(F)cc1N C(=O)(C(C)CCCCCC)N(CCOCCNC(C1(F)CC(OCC)C1)=O)C CC1CN(c2ncc(Cl)cn2)CCN1C(=O)CC(=O)NC1CCCCC1 c1(C(=O)NCC(F)CNC(c2ccc(CO)s2)=O)cc(F)c2cn[nH]c2c1 c1(OCC)ccc(N)cc1-c1cn(C(C)CNC(=O)Cn2cccn2)nn1 C12(C(=O)NCCC(C)NC(c3cnc(CCCC)s3)=O)CCC(C)(C1)OC2 N1(C(c2cc(C)c(C#N)cc2)C(=O)NC2CC2)CCn2nc3c(c2C1)CCCC3 N1(C(C(C(C)C)n2cncn2)=O)CCOC2(CCCN(Cc3cnco3)C2)C1 c1(C(CC)N(C(C2N(C(=O)OC)CCCC2)=O)C)cccc(Cl)c1Cl C1(c2n(CCC)nnn2)(Nc2cn(C)nc2SC)CCC2CN(C)CC12 CC(O)(CNC(C1(NC(=O)COCCCN=[N+]=[N-])CCSC1)=O)CCO C1(C(N(CC=C)C)=O)CC(C)CN(C(=O)Cc2cc(C)n(C)n2)C1 N1(C(CCc2c(C)nn(C)c2)=O)CC(NC(=O)C=C2CCC(C)C2)C(C)(C)C1 O=C(CCCS(=O)(=O)c1ccc(Br)cc1)Nc1cc(OCC(F)F)cc(F)c1 CCCCC(C)NC(=O)CCN(CCO)C(c1ccc(COC)s1)=O C1(C(N2CC(C)C(NC(=O)C(c3cc[nH]n3)C)C2)=O)CCC(C)(C)CC1 c1(NC(C2C(CNC(=O)CN3CCNC3=O)C2)=O)ccc(O)cn1 C1(C(=O)NCC(CC(F)(F)F)NC(CCCCC#C)=O)CN=C2N=CNN2C1 c1(NCc2cc(OC)ns2)nccc(=NC(C)c2ccc3c(c2)OCO3)[nH]1 c1(C(C(=O)NCC(CC)NC(=O)CN2CSCC2=O)C)cc(C)cc(F)c1 N1(C(c2[nH]cc(CC(C)C)c2)=O)CCC2(CC1)CN(C(=O)C(Cl)=CCl)CCO2 C1(C(N(C2CCN(C(=O)COC3(C)CCC3)C2)C)=O)CCc2nnc(O)n2C1 c1(CC(C)C)ccc(C(=O)NCCN(C(=O)C2=CCC2)C(C)C)s1 C1(NC(C=CC)=O)CCCCC1C(=O)NC1CCC=CCC1 N1(C(c2c(C)csn2)=O)CCCC(NC(=O)CN(C)CCO)CC1 C1(CC)CN(C(C2CC(=O)N2)=O)CCC1NC(c1n[nH]c(C(C)(C)C)n1)=O c1(N(C)C)cncc(C(N2CCCC2(C)CNC(=O)C(F)F)=O)c1 C1(C(=O)NC(C)C(=O)N2CCCC2)C=CCCN1C(c1ccc[nH]1)=O N1(C(Cc2nnn(C)n2)=O)CCCC(N(CCF)C(c2ccc(C(N)=O)cc2)=O)C1 N1(C(C(COCCCO)NC(=O)C(F)CC2CCOC2)=O)CC2C3CCC(C3)C12 CC1COCC(C(=O)N(CCCCN(C)C(c2ccn(CCF)n2)=O)C)O1 N1(C(C(CC)NC(=O)OC)=O)CCC(NC(=O)Cn2cncn2)CC12CCCC2 c1ccc(OC)c(OC)c1.c1(CNC(=O)OC)cccc(OC)c1.C1(=O)C(CC)N1 CC1CCCCC1CC(=O)N(CCC(=O)NC(C)(C)Cn1cccn1)CCO C(=O)(C(CCF)NC(=O)CCC1CCC(=O)C1)NCC#CCC C1(O)(C(C(=O)NCC2CC23CC3)NC(Cc2ncc(CC)[nH]2)=O)CCCCC1 C1(C(=O)NCC2C(NC(c3nnsc3-c3ccccc3)=O)C2)C2CC3C(C2)C13 c1(OC)cc(NC(c2nnnn2C2COC2)(C)CC2CCCCO2)cc(F)c1 c1(C(=O)NCCCN(C)C(C2(C#N)CC2(C)C)=O)ccc(Cl)c(F)c1 CC1CN(C(=O)C2=CCCS2)CC2(CCN(C(=O)C(C)(C)CS(C)(=O)=O)C2)O1 C1(CN(C(C2C(OC)CCC2)=O)C)COCCN1C(C1CCC(OC)CC1)=O CC(C)C(C)CC(=O)N1CCC(C)(C)C1CNC(C1CCCC1)=O O=S(=O)(c1ccc(=NCCN2CC3CC3C2)[nH]c1)N1CCC2(CC1)CC2CO Cc1cc(N)ccc1C(N1CCC(C)(C)C(NC(=O)CCC(F)F)C1)=O c1(C(=O)NCC2(C)N(C(CCC(CC)C)=O)CCC2)ccc2[nH]c(=N)[nH]c2c1 c1(NC(C2CCC(NC(c3cc(SC)nn3C)=O)CO2)=O)cc(O)c(Cl)cc1Cl c1(C(=O)NCC(CN(C)C(C2(c3cccs3)CC2)=O)(C)O)ccc(CO)cc1F CC1CCC(CCNC(C23CC(NC(=O)C(C4CC4)N(C)C)(C2)C3)=O)O1 N1(C(C(C)N(S(C)(=O)=O)CCOCC2CCCC2)=O)CCC(C(=O)OC)C(O)C1 C1(NC(C=CCOC)=O)CCCC(NC(=O)CNC2CCOC(CC(C)C)C2)C1 Cc1c(CN2CCC(CNC(C3CNC(=O)O3)=O)C2)cnn1C c1(NC(=O)CCCC2CC2)cnc2c(c1)CN(C(=O)CCc1nncs1)CC2 n1(CCOC)nc(C(=O)NCc2cn(C3Cc4ccccc4C3)nn2)ccc1=O c1(C(=O)NCC(C2CC2)NC(CCCC(=O)OC)=O)cc2c(ccn2C)c(O)n1 N1(C(c2c(C)cc(C)s2)=O)CCC(C)(C)C(NC(=O)CCn2ncn(C)c2=O)C1 Cc1cnc(C)c(C(=O)NC2CCOCC2NC(=O)CC2CCC(C)CC2)c1 N1(C(c2c(C)nc(N(C)C)s2)=O)CC(NC(c2cn(C)c(=O)n2C)=O)CC(C)C1 C1(C(=O)NCCN(CCCC)C)CC(NC(=O)Cc2cccs2)C1(C)C S(=O)(=O)(c1ccc(OCC(F)(F)F)cc1)NCC(CSC1CCC(C)C1)O C1(CC(=O)N(CCNC(=O)CC(C)C(C)C)CC)SC2=NCCN2C1=O N1(C(=O)Cc2csnn2)CCn2ncc(-c3cn(Cc4ccno4)nn3)c2C1 C(=O)(C(C)C(CC)CC)NC(CC#C)CC(=O)NCC(c1ccccc1)F C1(C(N2CC(SCCOC)C2)=O)CCCCCN1C(=O)CCOCC C=CCC(CC=C)C(=O)N1CC(C(=O)NC2CCCC2F)C(C=CC)C1 C1(C(=O)NC2(C)CC(C)(C)C2)CC2C=CC1N(C(=O)C(C)(O)C(F)(F)F)C2 N1(C(Cc2c(C)occ2)=O)CCCC(CNC(=O)CC(C)(C)C2CCCCC2)C1 CC1(C(=O)O)CCCCC1C(N1CCC(CCCF)CC1)=O Cc1cccc(C(=O)NC2CCCC2NC(c2cnn(C3CCOC3)n2)=O)c1C Cc1cc(C(=O)NC2(CNC(C3CCC4(CC4)C3)=O)CCOC2)c(F)cc1F N1(C(CCN(CCCC(C)C)CC)=O)CC(O)(C(F)C(=O)N(C)CC)C1 C(=O)(C1=CCC(C)(C)CC1)N(CC(C)O)CCNC(c1cnc2ccsc2c1)=O C1(NC(C2C(C)C2)=O)CCCC(NC(c2ccsc2COc2ccccc2)=O)C1 C(=O)(CC(F)(F)C(F)F)NC(CCCNC(C1C(C)CCOC1)=O)(C)C Cc1csc2c(N3CCC(CNC(C4CC5(CC(=O)N5)C4)=O)C(C)C3)ncnc12 C1(C)(C(=O)NC(CN(C(c2n(CCOC)ncc2)=O)C)C)CCCCCC1 C1(C2CC2)(C(=O)NCc2n(C(C)C)ncn2)CN(C(c2cncs2)=O)C1 c1(NC(C2CC3(C4CN(C)C4)C2C3)=O)ccccc1NC(c1ccccc1)=O C(C(C)(C)C(=O)N1CCCC(NC(c2c(C3CC3)cnn2C)=O)C1)SC c1(CC(=O)Nc2cc(F)c(C(=O)OC)c(F)c2)cc(Cl)c2c(c1)OCO2 N1(S(CC=C)(=O)=O)CCC2CN(C(c3ccc(SCC)s3)=O)CCC12 Cc1cccc2cc(C(N3CCC(F)(CNC(C4CCCC4O)=O)C3)=O)nnc12 C1(C(=O)NC(C2CCN(C(=O)C(F)(F)C(C)O)C2)C)Cc2cccnc2C1 Cc1nc(-n2cccc2)sc1CN(CC(C)(F)F)CC(C)C c1(C(=O)NCC(C2CCN(C(C(C=C)(F)F)=O)CC2)F)cc(C)c(F)c(C)c1 N1(C(c2n(C)c(S)nn2)=O)CC(NC(=O)Cc2cc(F)ccc2F)CC(C)(C)C1 C1(CN(C(c2scc(OC)c2)=O)C)CCCCN1C(C1COCC1(C)C)=O C1(NC(C2N(C(CC(C)C)=O)CSC2)=O)CC(=O)N(C2CCNCC2)C1 CC1(C(=O)NC2CCC2NC(C2(c3cccnc3Cl)CC2)=O)CCC(=O)CC1 C1(CNC(C2C(C(=O)OC)CC2)=O)CC(C(=O)N(C)CC2CCCS2)=NO1 CS(=O)(=O)c1cc(C(=O)NC2CC(NC(C3C=CC=CC=C3)=O)C23CCC3)co1 c1(SC)cccc(NCCCCNC(=O)C=Cc2ncc(C)[nH]2)c1[N+](=O)[O-] c1(NC(C2CCN(C(c3ccccc3S)=O)C2)=O)cccc2ccc(Cl)nc12 c1(C(N2C(c3cn(C(C4CCC4)OC)nn3)COCC2)=O)cnc(Br)c(I)c1 N1(C(CCc2nc(C)sc2)=O)CC2CC(C1)C2N=c1cc(Cl)nc(C2CCC2)[nH]1 c1(CC(=O)OC(C(CCOC(C)(C)C)C(F)(F)F)=O)ccc([N+](=O)[O-])c(N)c1 O=C(CS(=O)(=O)N1CCOCC(C2CCOCC2)C1)N=c1ccc(Cl)n[nH]1 c1(CNC(c2cn(CC=C)nn2)=O)ccc(CNC(C2(C(N)=O)CC2)=O)cc1 CCC(C)CC(C(=O)NCc1ccc(F)cn1)NC(C1CN(C(C)C)C1)=O C=C(CNC(=O)Cc1cnn(-c2ccccc2)c1)CCNC(C1CCC(F)C1)=O C1(C2(C)CC2)CCCN1CC1OCCC1C(=O)O C1(OC)C(C(=O)NCCCn2cc(-c3cc4occc4[nH]3)nn2)CC12CCC2 CC(C)CC(CNC(c1ccns1)=O)C(=O)N(C)CCN(C)C N1(C(c2c(C)scc2)=O)CC2CCC1C(NC(C1CC(C)C1C)=O)C2 c1(C(N(C2CCN(C(C3CCCOC3)=O)C2)CCC)=O)cncc2cccnc12 c1(C(=O)NC2(C(N(C)CC3C(C)C3)=O)CC(F)(F)C2)cncc2[nH]ccc12 c1(C(=O)NC2CCN(C(C(C(=C)Cl)(C)C)=O)CC2)[nH]c2cccc(F)c2c1Cl C1(NC(C2CCSC2)=O)CCC2CN(C(c3cnn4c3CCCC4)=O)CC2C1 c1(C(N2CC(NC(C=Cc3cnc(C)s3)=O)C3C2C3)=O)ccc([N+](=O)[O-])cn1 c1(NC2C(C)CN(C(=O)C(=O)NC3CC3)CC2C)nc2cc(F)ccc2o1 c1(CNC(N2CC(CN(C(C)C)C)OCC2)=O)ccc2c(c1)CCN(C)C2 C1(NC(c2c(CC)con2)=O)CC(OC)CN(C(C2CC2[N+](=O)[O-])=O)C1 c1(OCCOC)cc(C(=O)NC(C)C(C)NC(c2cncnc2O)=O)ccn1 C1(NC(Cc2nc(C(=O)OC)sc2)=O)CCCN(C(C2CC(F)(F)C2)=O)CC1 C1(C(=O)NCc2cc(C)sc2)CC(=O)CC12CCC2 CCC(C)(COC)CNC(=O)CCC(C)NC(C1CC1(Cl)Cl)=O c1(C(N2CCC(CC=C)(NC(c3coc(CO)c3)=O)C2)=O)nc(=O)cc(N)[nH]1 N1(C(C2C3(CCN(C(CSCC)=O)C3)C2)=O)CC2NC(=O)OC2C1 C(CCSC)(C(=O)NC(c1nccs1)(C)C)NC(C(C)OCC=C)=O CCC(F)C(=O)N1CC(O)(CN(C(=O)C(c2occc2C)c2cccs2)CC)C1 c1(C(=O)NC2C(O)CCN(C(C(P(C)(C)=O)O)=O)C2)ccc(F)c2cccnc12 c1(OC)cccc2c1OC(C(=O)OC(c1cc(F)c(NC(C)=O)cc1Cl)=O)C2 N1(C(C(CC)O)=O)CC2CC2C1C(=O)NCCc1ccncn1 N1(C(CCCOCC)=O)CC(NC(C2CNC(=O)N2)=O)C(C)(C)C1 C#CCC(C)(CC)C(=O)N1CCC(O)C(NC(C2CC2=C)=O)C1 C1(NS(N)(=O)=O)(CN)CCN(C(c2cncc(-n3cnnn3)c2)=O)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(=O)CC2CCCN2CC)C12CCC2 C1(C(=O)NC(CC(C)C)CNC(=O)CCCc2cccnc2)CCC(C)(C)CO1 c1(C(=O)Cn2cc(C(C)(C)NCC3CCCO3)nn2)ccccc1CNC(N)=O c1(NCC2N(C(c3ncc(Cl)cc3Cl)=O)CCC2)nc(Cl)[nH]c2ncnc1-2 N1(C(c2c(C)nc(C)s2)=O)CCOCC(C(=O)NCC(C)(C)c2cccs2)C1 C(CC(=O)N1CCC(N(C)C(c2ncc[nH]c2=O)=O)C1)(C1=CCCC1)OCC CCCC(CCCN(C(=O)OC(C)(C)C)C1CC1)NC(c1cc(C)on1)(C)C c1(C(N2CCC(NC(c3c(COC)n(C)nc3)=O)(CF)C2)=O)ccnc(Cl)c1O C1(N(C(=O)CCN2CCCC2=O)C)CC2CCC(C1)N2C(=O)C(=O)NC1CC1 c1(OC)cc(NC(C2CCN(C(=O)CN3CCSCC3)CC2O)=O)nc(Br)c1 C1(C(=O)NC2C(C)CN(C(c3cccc(Cl)c3)=O)C2)CN(C(N)=O)CCC1O N1(C(CC(CC)O)=O)CCCC(NC(c2cc(NC)nc(Cl)c2)=O)C1C c1(C(=O)NCC(CNC(C(C)CSC(F)(F)F)=O)(C)O)ccc(N)cc1F N1(C(c2c(CC)n[nH]c2)=O)CC2CC(NC(c3cn(CCF)nn3)=O)C(C2)C1 C1(O)(C(C)NC(c2cccc(N3CCCC3)n2)=O)CCN(C(=O)COCCF)C1 CC(C)(O)C(F)C(=O)NCC1CN(C(=O)C2=CCCCO2)CC1C(F)(F)F C1(COC)CN(C(c2sc(Br)nc2C)=O)CCN1Cc1ccc(OC)nc1 N1(CC(N2CC3C(C(=O)NC4CCC(C(=O)O)C4)(C3)C2)=O)CCn2ccnc2C1 c1(C(N2CC(CC(C)NC(C(CSC)O)=O)C2)=O)noc2ncccc12 COC1OC(=O)c2c(F)c(C(=O)OCc3nc(N(C)C)n[nH]3)cc(F)c21 Cn1ncc(C(=O)NC2CCN(C(=O)CCn3ccnn3)C2C2CC2)c1C1CC1 C1(CNC(C(C)SC)=O)CC2(CC2)CN1C(=O)CCN1CCCCC1 C1(C(C)C)CCC(C)CC1C(=O)NCC1(C(C)NC(C2(F)CC=CC2)=O)CC1 C1(NC(=O)CC2=CCC2)CN(C(=O)C=Cc2ccc(OC(F)F)cc2)CC12CC2 C1(NC(CSCC(C)C)=O)CC2CN(C(C3(F)C(C)(C)C3(C)C)=O)CC2C1 C12(C(=O)NC(C)(C)CCNC(=O)CSCCC(F)(F)F)CCC(C1)CS2 C1(CNC(C(C)C2CC2)=O)CCCN1C(=O)CCc1nc(O)n[nH]1 Cc1ccc(Cl)c(C(=O)NC(C)CCNC(=O)CCc2ccoc2)c1 C1(C2CN(C(C3(F)CCS(=O)(=O)C3)=O)C2)(NC(c2cccnc2O)=O)CC1 C(=O)(CCCCCCC(C)=O)NCC(CC=C)NC(C12CCCCC1C2(F)F)=O CCCC(CCC)CC(=O)N1CCC2(CCN(C(=O)CSCCC(C)C)C2)C1 N1(Cc2cc(OC)c(F)cc2)CC2C(C1C(=O)NC(CO)C(C)O)C2(C)C N1(C(c2ccc(CC)[nH]2)=O)CCN(C)CC1CNC(=O)C(c1c(C)noc1C)C C1(CC(=O)NCC#CCNC(C2C(CC)C2)=O)(CO)CCCC1 CC1(C)COCCC1C(=O)NCCC1(NC(c2cc(Cl)ccc2Cl)=O)CC1 c1(C(N2CCC(COC)(CNC(C3(Br)CC3)=O)C2)=O)cn(C)c(=O)n1C C1(F)(CNC(c2ccsn2)=O)CC(N=c2nc(CC3CC3)[nH]s2)C1 C(=O)(CC1=CCCCC1)N1C2C(CNC(c3c(CC)c[nH]n3)=O)C(C2)C1 C1(F)(C(N2CCC(CNC(C(C)c3ccco3)=O)CC2)=O)C(F)(F)C1(F)F CC1CC(CNC(C2(C)CCC2)=O)CN1C(c1cc(C2CCOCC2)[nH]n1)=O C(=O)(C(C)CC(=O)N(CCCCCNC(=O)C1CC1)C(C)C)OC Cc1ccc(CCC(=O)NCCCN(C(C2(CO)CC2(F)F)=O)C2CC2)cc1C c1(C(=O)NC2(CNC(C)=O)CC2)coc(C(F)F)c1 c1(C(N)=O)cc(CC(=O)NC2(CNC(C3CC34CCC4)=O)CCC2)cs1 CC(CCCCc1cccnc1)c1nccn1CC(F)(F)F N1(C(c2cnc(CC)[nH]2)=O)CCCCC(NC(c2cc(O)nc(C)n2)=O)C1 C(C(CC(=O)N(C1CN(C(C2(C)CCCS2(=O)=O)=O)C1)C)C(F)(F)F)N(C)C C=CC1CN(C(=O)C(CCSC)NC(c2ccc(C)c(O)c2)=O)CC1O CC(C(CO)NC(=O)CCCN(C)C)NC(=O)Cc1cnoc1 C1(CC(=O)NCC(CC)NC(=O)C(C2CCCCC2)O)COc2ccccc2O1 c1(C(N(CC(C)NC(Cc2c(C)noc2C)=O)C)=O)cnn2cnnc2c1 Cc1ccn2ncc(C(N3CC(C4(NC(=O)Cc5ccsc5C)CC4)C3)=O)c2n1 n1(CC(N2CCC(N(C(=O)CC3CC(SC)C3)CC)C2)=O)cc2ccccc2n1 c1(C(=O)NCCNC(c2c(NCC)scn2)=O)cc(C(C)C)oc1C N#CC1CCN(C(=O)C(C2CC=CCC2)NC(C2CCC3(CC3)C2)=O)CC1 O=C1CCC(CC(N2CCC(CCC(=O)NOCCCCF)(CF)C2)=O)CN1 c1(C(=O)NC2(C)CN(C(C3C(C)C3)=O)C2)cc(S(C)(=O)=O)ccc1F CCC(C)(CCC(C)C)C(=O)N1CCC(C(=O)NCCc2ccc(Cl)cc2)=C(F)C1 Cn1c(CC(N2CCOCC2CCF)=O)nc2ccccc12 CC1=C(C(=O)N2CC(N(C)C(c3cncc4ccsc34)=O)C3(CC3)C2)CCCO1 C1(NC(CC(C)OC)=O)CCCCC12CCN(C(c1cc(O)cc(=O)o1)=O)CC2 N1(C(C(C2CCCCC2)OC)=O)CCCCC1CN(C)C(c1cccc(N)c1)=O N1(C(C(=O)NCC(c2ccccc2F)(C)C)=O)CCOC2(CSC2)C1 c1(C(N2CCC(NC(=O)CNC(=O)C3CC3)C2)=O)csc2ccccc12 c1(C(=O)NCc2scc(C(=O)NCCCCCC=C)c2)ccnc(O)c1F C1(CC#N)CN(C(=O)C(Cl)(Cl)Cl)CCN1Cc1ccc(-c2ccccc2)s1 c1(CC(COC)O)cn(CCC(=O)N(Cc2ccccc2)Cc2nonc2N)nn1 N1(C(c2cn3c(n2)CCC3)=O)CCCC12CCN(C(C1(CO)CCOCC1)=O)C2 Cn1cc(Br)c2c(NC3CCCCC3c3cccc(Cl)c3)ncnc12 c1(SCC)cncc(C(N2CCC(N(C)C(C3(CC(C)C)CCC3)=O)C2)=O)n1 c1(OC)ccc(C(=O)NC(C2CCCCN2C(=O)CC2(OC)CC2)C)cc1N N#Cc1cc(CNC23CC(NC(=O)CNC(=O)CCCCO)(C2)C3)ccc1F N1(C(CCCc2onc(C)n2)=O)CCN(C2CN(C(C3C(C)C3C)=O)C2)CC1 N1(C(C2C(OCC)C2)=O)CCSCC1CCNC(=O)C(C)Cc1ccccc1Cl N1(C(CCSCCCC)=O)CC2(C1)CN(C(C1CC1CC)=O)C2 C1(OCC(=O)NC2CCN(C(C3CCN(SCC)CC3)=O)C2)C#CCCCCC1 CC(C)C(C)(O)C(=O)NCc1cccc(NC(C2CCN2S(C)(=O)=O)=O)c1 c1(N2CCN(C(=O)NCCc3ccc(SC)cc3)CC2)cncc2nnnn12 Cc1ccc2cc(CN3CC4OC(C)(C)OC4C3)[nH]c2c1 C1(CN(CCCCN(C)C)CC)CCN(C)CC1C CN1CCCC(CCC(=O)N(C)CCNC(=O)C(F)=C2CCC2)C1 C1(CN(C(c2nc(COC)oc2)=O)C)C2CN(C(=O)C(F)=C(C)C)CC12 C(=O)(CC(C)C(F)F)NC(CCOCC)C(=O)NC(C)Cc1nncn1C N1(C(c2scc(OC)c2OC)=O)CC(N(C(=O)C(C)SC(F)(F)F)C)C2(CC2)C1 C1(=O)C2n3ncc(-c4ncccn4)c3N1C2.C1CC1(C)C.CO C(CC(C)N=c1[nH]nc(C2CC2)o1)NC(c1cncc(COC)c1)=O C1(CNC(C2(COC)CCCC2)=O)C2CN(C(c3cc(O)no3)=O)CC12 C(=O)(CC1CCCN(C)c2ccccc21)NC1CCN(CC)CC1C C=CCC(C)(C)CCOCC(=O)Cc1cccc(OC)c1 C(CC(CC)C(=O)NCCn1cc(CNC(=O)COCc2nc[nH]n2)nn1)=CC Cc1cc(O)nc(COc2cccc(N(C)C(=O)NC3(C)COC3)c2)n1 N1(CC(=O)NCCN(CCOC)C(c2[nH]cnc2C)=O)CSCCSC1 N1(C(C2CN(C)C2)=O)CC(NC(c2cccc(SC(F)(F)F)c2)=O)CC1CO C=CC1(C(N2CC3CCC2C(O)C3)=O)CCN(C(=O)CCCC=O)CC1.OC CC1CC(NC(c2cnns2)=O)CN(C(c2c[nH]ccc2=O)=O)C1 c1(C(=O)NC2C(NC(C(COC)OC)=O)CCOC2)cnn2ccccc12 c1(C(=O)NCCOCCNC(=O)C2=C(Cl)CCC2)ccc(F)cc1F c1(C(N2CC=CC(NC(C(C3CCCC3)OC)=O)C2)=O)ccc2cn(C)nc2c1 c1(OC)ccccc1-c1c[nH]cc1C(=O)NCC(CNC(=O)CCF)OC c1(NC(C(=O)NCC2CC(SC)C2)=O)cn2ccc(Br)cc2n1 N1(C(c2c(OC)cccc2)=O)CC(NC(C2CC(C)OC2C)=O)CC2(CC2)C1 c1(C(=O)NC23CN(C(C4(CC=C)CC=CC4)=O)C(CC2)C3)ccc(F)cc1C#N C(=O)(CC(COC)NC(=O)COc1ccccc1)N(CC(=O)NC)C c1(C(=O)NCC2N(C(C3(COC)CC3(F)F)=O)CCC2)cc(C#N)n(C)n1 Cc1c(C(F)(F)F)n[nH]c1C(=O)NCC1CCN(C(C2CCSCC2)=O)C1 c1(C(N(CC(C)NC(C2C(C)C2(F)F)=O)CC)=O)nnc2ccccc2n1 C1(N(CC(c2cncn2C)(C)C)C)CCCN(Cc2nccs2)CC1 Cc1cc(O)nc(C)c1C(=O)NCC(C)NC(C1(C)CCCCO1)=O Cc1sc(-c2ccco2)nc1C(=O)NC1CCCC(CNC(c2cc[nH]n2)=O)C1 C#Cc1ccc(CC(=O)NCCN(C2CC2)C(c2ccc(C(C)F)cc2)=O)cc1 N1(C(c2ccc(C)o2)=O)CC2CCC2(CC(=O)NCCC2CC2C)C1 c1(C(=O)NC2CN(C(CCC=C)=O)CC2(C)C)cc2ccccc2cc1F N1(C(c2c(C)nc(CCC(F)(F)F)o2)=O)CCC2(NC(=O)CNC=O)CCCC12 C(=O)(CCCC(F)(F)F)NCC1(C)CN(C(C(C)=C(C)C)=O)C(C)(C)C1 C(=O)(CCCN=C1NS(=O)(=O)c2ccccc21)NCC(CO)NC(C(C)N(C)C)=O C1(C(C)C)CN(C(=O)C=CC2COC(C)(C)O2)CCN1C(C1CC(F)C1)=O C(C(CC)CCO)NC(C1(F)CC(NC(CCNC(=O)NC)=O)C1)=O C1(C)(C(N2CCCC(OC)C2)=O)CC12CCN(C(=O)CC(O)CC)CC2 C1(C(=O)NC(CNC(C(CC)N(C)Cc2ccccc2)=O)CO)CCN(C)CC1 Cc1c(CNC(=O)OC(C)(C)C)cccc1S(=O)(=O)N1CCOC2C(C(=O)O)C12 c1(C(N(C2CN(C(c3cc(C)sc3)=O)CC23CC3)C)=O)cc2cnccc2[nH]1 c1(CNC(C2C(NC(C3ON=C(CC)C3)=O)COC2)=O)[nH]ccc(=O)c1O C#Cc1ccc(C(=O)N(C(C)CCNC(c2c[nH]cc2CC)=O)C)c(F)c1 c1(CC(=O)NC2CC(NC(c3n(CC)nc(C)c3)=O)C2)c(O)ncnc1O C1(CNC(CCC)=O)CC(NC(=O)CCSCc2ccccn2)C1(C)C CCCC(F)C(=O)NCC1(CC(=O)N(CC(C)O)CCO)CC1 C1(NC(c2c(C#N)scc2)=O)CC(C(=O)NCC2CC3(CC3)C2)C12CCC2 c1(-c2n(CC(=O)NCCC=C)ccn2)ccc(-c2cccc(CC(N)C)c2)cc1 C(=O)(C1Cc2ccccc21)NC1C(NC(CCN(CC=C)C(C)=O)=O)CCC1 C(CCN=c1nc2c(cnn2C(C)C)c(NC2CC2C2CC2C)[nH]1)OCCCC N1(C(CC(C(C)C)C)=O)CCC2CCN(C(=O)CSc3cnn(C)c3)CC2C1 c1(C(C(=O)OC)NCCCCCSC)cc(C(N)=O)sc1C C(c1c(C)coc1C)=CC(=O)NC(CCNC(c1onc(CC)c1C)=O)C CC1=NN(C)C(=O)C1CC(=O)NCCCCCNC(C1(CF)CC2(CCC2)C1)=O Cc1cc(=NC(=O)C2CCN2C(C(C)CC(C)(C)c2ccccc2)=O)[nH]n1C c1(C(N(CCC)CCNC(=O)CCC2CC2C)=O)nsc2ccccc12 C1(O)(CC(=O)NCCCCn2ccnc2)CN(C(=O)Cc2cnc[nH]2)C1 N1(C(c2cc(OC)c(C)cc2)=O)CC2CCCN(C(=O)C(=O)NCCC(N)=O)C2C1 C1(C(=O)NC(C2CCN(C(Cn3c(C)nc(C)n3)=O)CC2)C)CCOCC1(C)C c1(CCC(=O)OCC(N(C)C)C2CC2)cccc(OC(F)(F)F)c1 CS(C)(=O)=NCCNC(=O)CC1CCCN1C(C1CCC2CC2C1)=O C1(NC(Cc2ncc(C)nc2)=O)CCN(C(=O)Cc2cc(C3CC3)no2)CC1C Cc1cc(C(F)(F)C(=O)NCC2(CNC(C3SCCC3C)=O)CC2)cs1 N1(C(=O)NC)CCC(C)(C(=O)Nc2cccc(NC(=O)C(C)(C)C)c2)C1 c1(CNCc2cn(CCCO)nn2)noc2c1CCCCC2 c1(N2CC3C(NC(=O)NCc4c(C)cccc4)C3C2)ncc2c(ccn2C)n1 c1(-n2ccc(C)n2)cccc(F)c1NC(=O)C(N1CCOCC(O)C1)=O N1(C(C(C)N(C(=O)CN(C)C)C2CCC2)=O)CCCC(C)(C)C1C C1(NC(c2[nH]nc(OC)c2Cl)=O)CCCCC12CCCN(C(C1CC=CC1)=O)C2 C(=O)(C1c2c[nH]nc2CN1C(C1CC2(C1)CC(O)C2)=O)N1CC(CC(=O)OCC)C1 C(=O)(CC(=O)NCC1(C(=O)NCCOC(F)F)CCC1)OC C(=O)(C(CNC(=O)CCCCN(C)C)CC(C)C)NC(c1nc(C)on1)C C1(NC(C(C)CN(C(=O)CCc2cn(C)nn2)C2CC2)=O)CCCC1(C)C C(=O)(C1=CC(O)CCC1)N1CC(CCCNC(c2cscc2C2CC2)=O)OCC1 CCCC(CC)C(=O)NC1CCC(C2CC2)C1.C(=O)(NOCCCC)C1(C)CC1 C1(NC(c2ccc(OC)c(I)c2)=O)C2CCC1CN(C(=O)CS(N)(=O)=O)C2 c1(N2CCC(F)(CNC(C3OCC(C)C3)=O)CC2)ncc2ccsc2n1 c1(C(=O)NC2CCN(C(CN(CC)CC)=O)CC2O)ccc(F)c2ncccc12 N1(C(CC2N(C)CCCC2)=O)CCC(C2CN(C(C3(C)CC=CCC3)=O)C2)CC1 N1(C(c2ccc(CC)cc2N)=O)CCC2(CC1)CN(C(C1CCC(OC)C1)=O)C2 C1(C(N2CC(NC(=O)C=CC3CCCCC3)C(O)C2)=O)C2CCC(F)(F)C12 C1(C(=O)NCC2CCN(C(C(C)OCC(C)C)=O)C2)CCc2nccn2C1 CC(=NO)C1CC(C(=O)NC2CCCCCN(C(=O)C#CC3CCC3)C2)C1(C)C c1(C(=O)OC)[nH]c(=NC2CC3CN(C(C4CC(C(C)C)=NO4)=O)CC23)sc1C C1(=O)C(CCCl)NC(=O)CN1CCOC(C)C.C(CCN)N.C(C)(=O)OCC.CO Cc1n[nH]c(=NCC2CN(C(c3csc(C4CC4)n3)=O)C2)s1 C1(NC(Cc2n(C)nnc2)=O)C2CCN(C(c3ccc4c(c3)OCO4)=O)CCC12 C1(NC(c2cnc(C(C)C)[nH]2)=O)CC(OC)CN(C(c2sccc2C(C)=O)=O)C1 c1(C(=O)NCCNC(c2cncc(C(C)C)c2)=O)cccc(P(C)(C)=O)n1 C1(CNC(c2cncc(CO)c2)=O)C2CN(C(c3cc(O)no3)=O)CC12 N1(C(=O)C(c2ccccc2)c2ccccc2)CCS(=O)CC1C1CCC1 c1(OCC(N2C(CC)CCC2)=O)cccc(C)c1 C1(OCC)CC(N(C)N2CCC(N3CCCC3C(N)=O)CC2)C12CCC2 C#Cc1ccc(Cl)c(C(N2CCC(C3(NC(=O)C(C)COCC)CC3)C2)=O)c1 Cc1cc(C)nc(N2CCC(C(=O)NC(=O)CCc3ncc(Br)cn3)C2)n1 C(CC(C)(C)C)(c1ccc(F)cc1)NCC1N(C(=O)OC(C)(C)C)CCC1 N1(C(Cc2c(C)n[nH]c2)=O)CCN(C(=O)CN2CCC(C(N)=O)CC2)CC(O)C1 C1(C(N2CCC(CCNC(c3cn(C)c(O)n3)=O)C2)=O)OCC2CCCCC12 C#Cc1cc(F)c(C(=O)NC2CC(C)(NC(C3CCC(C(N)=O)C3)=O)C2)c(F)c1 C(=O)(C(C(C)OC)NC(=O)Nc1ccccc1OCc1ccc(Cl)cc1)OC S(=O)(=O)(c1cccc(C(=O)NCc2n[nH]c(=N)o2)c1)N1CCN(CC(C)O)CC1 c1(C(=O)NC2CC3CN(C(C4(C)C=CCCC4)=O)C2C3)cnn2cccc(Cl)c12 c1(C(=O)NC(c2cccc([Si](C)(C)C)c2)C)cnc2c(cnn2C2CCCC2)c1 C1(C(=O)NCC=CCNC(C(=O)NCCOCCCC)=O)(SC)CC1(F)F c1(OC)cc(Br)ccc1CNCC1CCCN(C(c2cc(Br)ccn2)=O)C1 c1(NC(=O)NC(CC(C)=O)C)c(F)cccc1Br CC1CCC(NC(=O)C(F)=CC2CC2)CN1C(=O)COc1ccccc1 N1(C(c2cccc(NC)n2)=O)CC2(C1)CN(C(C1CC1c1ccccn1)=O)C2 C12(CNC(C(C3CN(C(C4SCC(=O)C4)=O)C3)O)=O)CCC(CC1)OC2 C1(CCNC(Cc2nc(C)[nH]n2)=O)C(C)CCCN1C(c1cnnc(O)c1)=O c1(OCC)c(F)c(C(N2CCN(C(=O)C(C)C)C3(CCC3)C2)=O)cc(F)c1F CCC(CC)CCC(=O)NC1CC1CNC(=O)CN(c1ncnc2[nH]cnc12)C C(c1ccc(F)cc1)=CC(=O)NCCN(C(c1ccnn1CCF)=O)C1CC1 N1(C(C2(CCNC(=O)CC(O)C3CCCC3)CCC2)=O)CC2C=CCC(C2)C1 C1(CC(=O)N(CC(C)(C)C2CCCO2)C)CCCCN1C(C1CC12CC2)=O c1(N2CC(CN(C)C(C3CCN(c4nccs4)CC3)=O)OCC2)cnc(C#N)cn1 CN1Cc2ccccc2C1CNC1CCc2ncsc2C1 c1(C(N(CC(C)NC(C2(CC)CCCO2)=O)C)=O)cc2sc(C)cc2[nH]1 N1(C(c2cnn(C3CC3)c2)=O)CCC2(CCCN(C(C3CC4(CC4)C3)=O)C2)C1 c1(CN(C(c2cnc(C3CC3C)s2)C(=O)NCC)CC)ccc(C#N)cc1F CCC(CC)(CC)C(=O)N(CC(O)CNC(c1nccc2cc[nH]c12)=O)C c1(NC)ccc(C(=O)NC2CCC2NC(C2(c3ccc(F)cn3)CC2)=O)cc1 C(N=C(NC1CC1C)N1CCOC2(CCCCC2)C1)C1CCC(C(=O)OCC)O1 N1(C(CCCC)=O)CC(C2(NC(C3(Cc4ccc(C)cc4)CCCC3)=O)CC2)C1 N1(CC(=O)N(CCN(C(CCN(C)CCO)=O)CCF)C2CC2)CCCNC1=O C=CCCN=C(NCC12CC1(C)C2)N1CCC(CCOC)C1 C#Cc1c[nH]nc1C(N1CCC(N(C(=O)C=Cc2scnc2C)CCO)C1)=O C1(NC(c2c(C)cno2)=O)CN(C(c2ccc3cnsc3c2)=O)C2(CCOC2)C1 Cc1ncc(C=CC(=O)NCCCCC2CCCN(C(C3OCCO3)=O)C2)s1 C1(NC(C2(CC#C)CCOC2)=O)CCN(C(c2sc(CCC)nc2C)=O)CC1C C1(C(=O)OC)CC1C1CCN(C(c2cccc3o[nH]c(=N)c23)=O)CC1 N1(C(CCCN(C(C)=O)C)=O)CC(CNC(c2cn(C)cn2)=O)CC1C C1(C)(C(N2CC(O)(CCNC(C(CC)SC)=O)C2)=O)CC(C(C)C)=NO1 C=C(F)C1(CC(=O)NC2CN(C(c3nccnc3CC)=O)C2)CCC1 c1(CNC2CCC(NC(=O)C=CCBr)C2)cc(Br)cc(F)c1F C1(O)(CC(=O)NC(C(=O)OC)CO)CCN(C(=O)CCCc2sccc2C)CC1 c1(OC)cc(NC(=O)CC2CC3(C2)CN(Cc2ncc(F)cc2C)C3)cc(Br)n1 C(=O)(C1=CCCOCC1)N(CC(C)C(=O)NC(c1nccn1C)C)C C1(CCC(=O)OC)CN(Cc2ccn(-c3ccc(Br)cc3)n2)CC12CC2 c1(CC)cc(C)c(C(=O)NCCCNC(C2(CC(F)(F)F)CC2)=O)o1 C1(C(N2CCC(O)CC2)C(=O)NCCOC)CC2C(C1)C2(F)F.c1(SCC)cc(C)no1 n1(CC(=O)N(CCC(C)NC(=O)CSc2nncs2)C)c(O)nc2ccccc12 C1(C(=O)NCC(N2CCCC2)C)CN(C(c2ccc3c(c2)CC3)=O)C2(CCC2)C1 N1(C(C2CCN(C(N)=O)CC2)=O)CCCC(NC(c2ccc[nH]2)=O)CC1 c1(C(=O)NC2CN(C(C3C(OC)C3)=O)CC2C)cc2sccc2[nH]1 N1(CCC(=O)NCCN(C(C2(O)CC2(C)C)=O)CC)CCOCC1=O c1(C2C(NC(C(C3CN(C(=O)Cc4cnc(C)o4)C3)OCC)=O)C2)cccnc1 c1(CNC(c2cc(OC)c(Br)cc2OC)=O)cn(C)c(=O)n(C)c1=O Cn1c(=O)oc2c(C(N3CCN(C(C4CCC(C)(C)C4)=O)CC3)=O)cccc12 C#CCC(CC#C)C(=O)N1CCC(CN(C)C(C2COC(=O)N2C)=O)C1 Cn1nc(C(=O)NC2CCC(CNC(=O)CC3CSC3)C2)c2cc(F)ccc12 n1(CCC(=O)NCC(CC=C)NC(=O)CCC=CBr)cccnc1=O CCC(COC)C(=O)N(C(C)C(=O)NC(c1ccc(C)o1)CC)C C1(N(C(=O)C(F)C2CCOC2)CC)CCN(C(=O)CNC(=O)OC)CC1 c1(COC)ccc(SC(C2CN(C(=O)Cc3ccccc3)C2)C)cc1 C1(C(N2C(C)(C)C(CNC(=O)C3=CCCOC3)CC2)=O)CCC2(CCOCC2)O1 C=CCCCC(C(=O)NOCC)NC(=O)CCC(=O)NC1CC1 c1(C(=O)NCC2OCCN(C(C3ON=C(CC)C3)=O)C2)ccc(C)c(S(N)(=O)=O)c1 C(=O)(CC(C)C(F)F)N1CCCC(C2N(c3nnc(C)o3)CCC2)C1 c1(NC(C2CCC(CNC(C3CC4C=CC3C4)=O)CC2)=O)c(Br)ccc(F)c1F n1(CC2CC(NC(C3CC(SC)C3)=O)C2)nnnc1C(C1CC1)CN(C)C N1(C(CCCC#CC)=O)CCC(N=[N+]=[N-])(C(N2CCC(CCOC)C2)=O)C1 C(=O)(C(CO)C(C)(C)C)N1C(CCC)CN(C(=O)C(=O)NCC(F)F)CC1 Cn1cc(C(N2CCCCC2C(=O)NOCC2(C)CCC2)=O)ncc1=O CCC(C)CCCC(=O)N(C1CCC(NC(=O)CC2=CCCC2)CC1)C C=CCCC(O)CN(C)C(c1ccn(CCNC(C2OCCO2)=O)c1)=O C12(CNC(C(C=C)(C)O)=O)CCC(CN(C(c3cn(C)nc3O)=O)C1)C2 C(CC(C)(C)CC(=O)N1CC(O)CC1(C)C(=O)Nc1cnn(C(F)F)c1)OC C(=O)(CCC(C)(C)C(=O)NCCC1CCN(C(=O)Cn2nccn2)C1)OC C1(C(C)NC(=O)C(F)=C2CCCC2)CCN(C(C2CC2c2cncn2C)=O)C1 N1(C(C2C(C)(CC)C2)=O)CCC(n2cc(CNC(=O)CNC(=O)NC)nn2)C1 N1(C(C(C2CCOCC2)C)=O)CCC(NC(c2ccsc2C(F)F)=O)C1(C)C c12ccc(s1)S(=O)(=O)NC2.C(CC(C)CCNC(=O)CNC=O)NC(C(C)C)=O C1(C(=O)NC(C)C(C)(C)C)CCCCCC1NC(=O)C(C)(C)CC#N c1(C(N2CCCC(N(C(=O)C(F)CC3CCC3)C)CC2)=O)nc2c(s1)COCC2 C1(OC)CCCC12CCN(C(=O)C(F)F)CC2.C12CN3CCCC3(C1)C(=O)N2 CC1CC(C(=O)Nc2ccccc2-c2ncc[nH]2)CCS1(=O)=O CCC(F)(C(=O)OC)C(=O)N1CCC(Cn2cc(-c3cccc(CO)c3)nn2)C1 CCCCC(C(=O)NCCc1cccc(Br)c1)N1CCCC1C(=O)OC(C)(C)C N1(C(C(C(C)C)=O)=O)CC2(C(=O)N(C(C)CN(C)C)C)CC1CCO2 C1(NC(C(CC)(C)O)=O)CC2(C1)CN(C(=O)Cn1ncc(O)nc1=O)C2 C12CC3(C1)CC(C3)NCc1ccc(Cl)c(c1)C(=O)N2.n1(C(C)(C)C)cccn1 N1(C(CC#N)=O)CCCC(C2(NC(c3noc4c3CCCC4)=O)CC2)C1 C1(CNC(=O)C=Cc2ccco2)(CO)CCOCC1.C12CC1NC2=O.C1(=O)CN1 C1(F)(CNC(c2cc(CC)sn2)=O)CCN(C(=O)C(C)C2CCCC2)CC1 CCC(C(=O)N(C1CCCN(C(c2ccc(C)cc2C)=O)C1)C)C(C)(F)F C(=O)(C(F)C(F)(F)F)NC1(CCCCNC(C2CSCCS2)=O)CC1 C1(c2nc(-c3ccc(OC)cc3)nn2CCCN2CCCC2=O)CC2(CCC2O)C1 CCC(C)(COC)C(=O)NCC(C)(O)CNC(=O)CSC(C)C CN1CCc2ccc(C(=O)NC3CC4CC(C3)N(C(=O)Cc3ccns3)C4)cc21 N1(C(C(COC)O)=O)CCC2CCC(C1)N2C(C1(c2ncco2)CCC1)=O N1(C(C2N(C)CSC2)=O)CCC(C(C)(C)NC(C2CC(F)(CO)C2)=O)CC1 C(=O)(C(CCC1CC1)NC(=O)Cc1c(C)noc1C)NCC(C)SC C1(C(=O)NC2C(CNC(c3coc(Cl)n3)=O)CCC2)CCC2(CCC2)CC1 C(=O)(CC(C)C(C)(C)C)NCC(C)N(C(CC(CC)CC)=O)C c1(C(=O)OCC)cc(C(C)N(CCC(F)(F)Cl)C(=O)OC(C)(C)C)nn1C c1(OC)cc(-c2cn(C3CC(NC(c4cc(Br)ccc4Cl)=O)C3)nn2)ccc1F C1(NC(C)CNC(=NCCF)NCOC(C)(C)C)CCC2(CC1)CC2(F)F C(=O)(C(C(C)(F)F)c1ccccc1)NCC(C)(C)NC(C1C=CCCC1)=O N1(C(C=C2CCC(C)CC2)=O)CCC(NC(=O)CCC2(C)CC2)CC1C c1(C(N(CC(C)NC(=O)Cc2cnsc2)C2CC2)=O)ccnc(OC2CCC2)c1 CC(F)(F)C(C)(C)CC(=O)N1CCOC(CNC(c2cnc(Cl)[nH]2)=O)C1 N1(C(C(C)=C2CC2)=O)CCCC(CCC(=O)NCCC2CC3C=CC2C3)C1 C(=O)(C(C)(C)C(O)CC)NCC1N(C(CC=CCC)=O)CCCC1 C1(NC(C(C)=C(C)C)=O)CCN(C(c2ccc(-c3ccccc3)nc2)=O)C(C)C1 C1(C(N(CC(COC)O)C)=O)CCCCCCN1C(=O)C(C1CC1)C1CC1 c1(C(N2C(CNC(CCOCC)=O)CC(F)C2)=O)cc(OC)cc(OCC)c1N c1(C(=O)NC(C2(O)CCN(C(Cc3c(C)cco3)=O)C2)C)cc(C#N)ccc1C CC(C)C(C(C)NC(=O)CNC(c1cccs1)=O)NC(=O)CCCC#N n1(CSCCS(=O)(=O)NCc2cn(CCCC(=O)N(C)C)nn2)ccc([N+](=O)[O-])n1 Cc1ccc(C(=O)NCC2CC2NC(c2cc(Cl)cc(F)c2N)=O)c([N+](=O)[O-])c1 CC(N=c1[nH]c(=N)[nH]c(=NCCc2cnn[nH]2)[nH]1)c1ncc(F)cc1F c1(C(N(C(C)CNC(c2cn(C)cn2)=O)C)=O)cccc2oc(=N)[nH]c12 c1(C(N2C(CC(N3CC(COCC)C3)=O)CCC2)=O)ccc(CC)nc1 Cc1cccc(NC(=O)CSC(C)C(=O)N(C)C)c1 C(=O)(CS(C)(=O)=O)NC1(CO)CCC1.C(=O)(C(C)C)NCC(=O)OC(C)(C)C c1(C(N2C(CNC(COc3cn(C)nc3)=O)CCC2)=O)cnn(C)c1C#N S(=O)(=O)(c1cccc(Br)c1F)NCC1N(C(c2c(OC)nccn2)=O)CCC1 Cc1nc(Cl)[nH]c(=NC2CCCCC2NC(=O)C(F)(F)C(F)F)c1[N+](=O)[O-] N1(C(c2ccn(C)c2)=O)CC2(CC(NC(C3CC4C=CC3O4)=O)CO2)C1 C1(NC(c2c(C#C)c[nH]n2)=O)CCCC2CN(C(=O)CCN3CCOCC3)CC12 c1(NCC(CCCC)NC(c2nnn(C(C)(C)C)n2)=O)ncn(C)c(=O)c1Br C=C(C)CN=C(NCc1ccnn1CCC)N1CCc2ncsc2C1 c1(C2CCC(O)C2)ccc(F)cc1Cl.Cc1ncsc1C(=O)NCCCN1CC1 c1(NC(c2cc(OC)ncn2)=O)cccc(SC(F)(F)F)c1C CN1N=C(CC(=O)N2CC(C)(C)CC2C(=O)NC2CC(C)(C)OC2=O)CC1=O N1(C(c2cnc(C3CC3)s2)=O)CCC2C(CCCN2C(=O)CCC2CCCO2)C1 c1(NCCN(CCOCC)C)ncccc1S(=O)(=O)NCCc1ncnn1C c1(C(N2C(CC(=O)NC3(c4nc[nH]n4)CC3)CCC2)=O)ccc(O)cn1 CC(C)CCC(=O)C(=O)N1CCC1CNC(c1cccc(F)c1)=O N1(C(C(C)CC2CCC2)=O)CC(C2CN(C(C34CC(COC)(CO3)C4)=O)C2)C1 CS(=O)(=O)c1ccc(C(N2CCC3(CC2)CC3NC(c2cnc[nH]2)=O)=O)s1 N1(C(C2(C)COC2)=O)CCOC(CNC(c2cccc(C(C)(C)C)c2)=O)C1 C1(N(CCC(=O)N(CC(C)C)CCO)C)CC=CC(n2cnnc2)C1 C1(NC(=O)Cc2c(Cl)cccc2Cl)CCCN(C(C2CC=CC2)=O)CC1 C1(C(N(CCNC(C2C(C#C)C2)=O)Cc2ccccc2)=O)CCOCC1C c1(C(=O)NCC(C2(OC)CC2)O)cc2ccc(F)cc2nc1O C1(C(=O)NCCC(C)CCNC(=O)C(C)(C)CC(F)F)CCCC2(CCC2)O1 C(C(=O)N1CCCC1C)(C(C)C)NC(c1nc(CCC)oc1)=O C1(CNC(=O)COCCF)CN(C(c2cncs2)=O)C2(CCC2)C1 c1(CC(=O)NCC(NNC(=O)c2ccc(C)cc2)=O)c(C)nc2n1CCCC2 C(=O)(CC(CC)NC(=O)COCCN1CCCC1=O)N1CC(CNCC)C1 C(=O)(C(C)(C)C)NCCC(=O)NCC1C(NC(CC2CC(=C)C2)=O)C1 S(=O)(=O)(c1cccnc1Cl)N1C(C(N(CCOC)C)=O)CC(O)C1 c1(-c2cnc(C(N3C(C(N)=O)CC(F)(F)C3)=O)nc2)ccc2c(c1)OC(F)(F)O2 c1(N2CC3CC(=O)NC3C2)nc(=NCC2CCSC2)[nH]c2ccsc12 c1(C(N2CCCC(N(C(=O)C(C)CSC)CC)CC2)=O)cc(C)c(F)c(C)c1 c1(C(=O)NC2CC(CC(=O)NCC(CC)(C)O)C2)ccnc(NC)n1 C1(NC(c2ccc(CN3CCC(CS(C)(=O)=O)CC3)cc2)=O)CC2OC1CC2O N1(CC)CCOC(C(=O)NCC(CNC(c2ccnc(C(F)(F)F)c2)=O)CO)C1 C(=O)(C(O)CCCNC(=O)Cn1ccnc1)NC1(C(N)=O)CCOC1 c1(SC)cc(C)c(C(=O)NCC(C2(O)CCN(C(=O)CCc3cnoc3)C2)C)o1 C1(CCC(=O)N(C)NC(CCSCCOC)=O)CCCOC1.C12(CC1)CO2 c1(C(=O)NCC(CNC(C(P(C)(C)=O)O)=O)O)c(F)cc(F)c(O)c1F c1(C(=O)NCC(C)NC(CS(=O)(=O)NCC)=O)cccc(C)c1N CC1CCN(CC(=O)NCc2c[nH]nc2C2CCN(C(=O)CSC3CC3)C2)CC1 C1(C(=O)NCc2c(C(N3CCC(CC(N)=O)C3)=O)con2)CC(C2CC2)=NO1 Cc1[nH]nc2ncnc(N3CCC(CCNC(=O)C(F)CC4CCCCC4)C3)c12 c1(C(=O)NCC2CCC2NC(C2CC3CCC(C2)O3)=O)cc2cccc(Cl)c2s1 c1(C(N2CCN(CC(=O)Nc3c(C(=O)OC)nsc3)CC2)=O)ccc(Cl)cc1F C1(c2n(-c3cc(C)c(Cl)cc3)nc(CCO)n2)CCN(S(=O)(=O)N(C)C)CC1 C1(N(S(=O)(=O)CC)CC(F)(F)F)COCC1n1cc(C2(O)COC2)nn1 C(CN=c1[nH]c(=NCc2ccns2)[nH]c2c1CCC2)OCC(F)F c1(C(N2CCCC(CN(C(c3cc(OC)ncc3)=O)C)C2)=O)cccc(C)c1C c1(C(CCOC)NC(C2CCNC2c2ccccc2)=O)ccccc1C N(C1CC2(CCCC2)c2ccccc21)C(N1C(CCCC)CCC1)=O c1(NCC23N(C(C=CCOC)=O)CCC2CC3)cccc2ncccc12.C1CO1 c1(C(=O)NCCC(C)NC(c2cc(SC)oc2C)=O)cc(F)cc2nccnc12 C1(CC(=O)NC2CN(C(=O)COC3CCCC3(F)F)C2)CC2(CCC2)C1 c1(C(=O)NC23CCCC(NC(CC(C)F)=O)(C2)C3)cnc2nccn2c1 CCCCC(O)C(=O)NC12CC(C1)N(C(=O)C(C)NC(=O)NC)C2 c1(CC(N2C(C(=O)NCCCC(C)(C)C)CCCC2)=O)cccc(Br)c1F CN1CCN(C(=O)CCn2cc(C3COCC3O)nn2)C1=O CC1(C)COC(C)(C(=O)N(CCCNC(=O)CCSC(F)(F)F)CCO)CO1 c1(C(=O)NCC(=C)F)oc(CNC(=O)CC(C)C2CCCO2)nc1C C(=O)(C(CCC1CC1)NC(C1CC=CCC1)=O)N(CC(C)C)C1CC1 C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NCC(CNC(C(CC)C)=O)O N1(C(C(n2cc(Cl)cn2)C)=O)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C(F)C1 Cc1ccc(C(=O)NC2C3CCC2N(C(c2cc(Cl)cc(Cl)c2)=O)C3)c(C)c1 N1(C(CNC(CC(C)(C)C)=O)=O)CC2CCC(C1)N2Cc1cc(O)nc(O)n1 C(=O)(CC(CC#C)NC(c1oc(C)nc1C)=O)NC1C(CCC#C)OCC1 CS(=O)c1cccc(C(=O)NC2COCCC2NC(c2nocc2C2CC2)=O)c1 C1(CNC(c2c(C(C)C)ccs2)=O)COCCN(C(c2cccc(CF)c2)=O)C1 C#Cc1cncc(C(N2CCN(C(=O)COCC3(F)CC3)C(C)C2)=O)c1 N1(C(C(C)OCC=C)=O)CCC2CCCC(C1)N2C(=O)CSc1ccccc1 C1(C)(CNC(C(C2CN(C(c3n(C)ccn3)=O)C2)O)=O)CC(C)(C)C1 C1(NC(CC2CCCC(C)C2)=O)CCN(C(c2ccccc2F)=O)CC12CCC2 c1(SCC(=O)N(C)CC2OCCN(C(COC(C)C)=O)C2)ccc2c(c1)CCC2 C1(NC(CC(=O)N(C)C)=O)CC2CC1N(C(=O)C(C)(C)C)C2 c1(C(N2CCCC2CNC(C2CC2Cl)=O)=O)cccc(C(F)(F)C(F)(F)F)c1 CC1CC(CNC(=O)COc2ccccn2)CCS1 C1(C(=O)NCC2CC(OC)CN2C(C2CCCC2(C)C)=O)CS(=O)(=O)CC12CC2 C1(C(=O)NCC(C)OC(F)F)(CNC(c2cnc(O)o2)=O)CC12CCC2 Cc1cccc2c(C(N3CCCC4C3CCN4C(=O)C3=NNC(=O)C3)=O)csc12 C123CCC(CN(C1)C(C1C4CCCC14)C(=O)NC2)C3.Nc1ncccc1C(=O)O C(=O)(C(C)(C)C(C)(F)F)N.C1(OC(=O)NC)CCN(C(=O)C(F)CC2CCOC2)C1 C1(C2CCCO2)(C(=O)NC2CN(C(c3cccc(C#C)c3Cl)=O)C2)CCCO1 c1(NC(c2c(OCC=C)cccc2)C)cc(C)nc(C)n1 C1(CNC(C(C2CCCC2)OCC)=O)CCN(C(=O)CCc2ncc(C)[nH]2)C1 Cc1cccc(CN(c2cnn(CC3CCCO3)n2)Cc2cccnc2Cl)n1 C12(C(=O)NCC3(CC)CCC3)CC(CO)(CN1C(c1ccc(F)c(C)c1)=O)C2 c1(NCc2cc(C(=O)O)cc(Cl)c2)c(Br)cc(C(F)(F)F)cc1Br c1(C(N2CCN(C(C(C)(C)C)=O)CC2CF)=O)ncn2c1CCCC2 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N(C1CCN(C(=O)C(F)=C2CCC2)C1)CC N1(C(c2scc(C)c2C)=O)CC(CC(=O)NC2CC(C)(O)C2)CC1(C)C c1(CC)[nH]c(=N)sc1C(=O)NCC1(CNC(c2cnc(C)nc2)=O)CC12CCC2 c1(OCC(=O)NCC=C2CCN(C(C3C(C(C)C)C3)=O)CC2)ccc(F)c(F)c1 C=C(C)CCC(=O)N1CCC(N2CCN(C(C3CC4CC4N3C(C)=O)=O)CC2)C1 N1(C(CC(c2c(C)noc2C)C)=O)CC2(CCCN(C(C3(F)CCCC3)=O)C2)C1 C=CCN=C(NCCc1ccn(C)n1)N1CCCC(S(=O)(=O)N(C)C)C1 CC(C)C(C)CCNC(C1C2CN(C(=O)C(c3cncnc3)C)CC12)=O N1(C(C2N(C(C)=O)C(=O)CC2)=O)CCC2(CC1)CN(C(C1(C#N)CC1)=O)C2 N1(c2ncnc(NCC(=O)NC)c2C)CCOCC2(COCCN2C)C1 N1(C(c2ccc(C)cc2)=O)CCC2(CCCC2C(=O)Nc2ccc(C#N)cc2)C1 CC(C)C(O)C(=O)NC.C12(C)CN(C1)C(=O)C(C1CCN1C(=O)OC(C)(C)C)N2 Cc1cc(C(=O)NC(C2(O)CN(C(c3sncc3C)=O)C2)C)nc(O)c1 C1(CNC(CCNS(CC)(=O)=O)=O)CC2(CCC2)CN1C(=O)Cn1cncn1 C1(CC)CCN(C(C2CCCC(=O)C2)=O)C(C(=O)NCc2ccsn2)C1 C#CC12CCC(C(N3CC(CNC(c4scc(C)c4Cl)=O)C3)=O)(CC1)CC2 Cc1cc(P(C)(C)=O)oc1C(N1CC2CC2(NC(c2cc(N)cnc2Cl)=O)C1)=O C1(C(N2CCCC(OC3CC3)C2)C(=O)NCNCCO)CCCCCCC1 C(c1ccc(C2CC2)cc1)=CC(=O)NC1C(N(C(C2C(OC)C2)=O)C)CCCC1 N1(CC(C)NC(=O)COC2CCN(C(C3COCOC3)=O)C2)CCCCC1 c1(N(C)C)ncnc2cc(CNc3cnc(Cl)nc3)ccc12.C123CC(C1)(C2)CN3 CC1C(=O)CCC1C(N1CCC(CC(=O)NC2CCC(N(C)C)CC2)CC1)=O CCCC(CNC(c1oc(CNC(c2[nH]ccc2C2CC2)=O)cc1C)=O)CCO C(CC(C(C)C)NC(=O)C(CNC(=O)COCCCCC)CC1CC1)OC C1(CNC(C(C)C)=O)COCC2(CCCN(C(=O)C(C)SC3CCCC3)C2)O1 C1(CNC(=O)CCC2CCCO2)COC(CNC(c2nc(CC3CC3)cs2)=O)C1 CC1=NOC(C(=O)NCC(O)CCNC(=O)CCOC2CCOCC2)C1C C(=O)(C(CNC(=O)NCc1nnsc1C(=O)OC(C)(C)C)O)NCC.OC CCCCCC(=O)N1CC(C(=O)NCC(N2CCC(C(F)F)CC2)=O)C1 c1(OCC)nc(N2CC(C)(C)CC2CNC(=O)CSSC)ncc1C O=C1OC(C(=O)NC2COC3(C2)CN(C(=O)CCC(F)F)C3)Cc2ccccc21 C(CCC)(CCC)=CC(=O)N(CCN(C(C(CC)=CC)=O)CC)CC c1(CC(N2CCC(NC(CC(C)SC)=O)(CF)C2)=O)ccc(Cl)c2cccnc12 C(=O)(C#CC1CCCCC1)NC(CC=C)CNC(=O)Cc1cncnc1 C12(C(=O)Nc3cncc(CO)c3)CCC(CC1NC(c1cc(C3CC3)on1)=O)C2 C(CCCCC(=O)N1CC(NC(=O)NC)C1)N(C(c1cccc(CC)n1)=O)C CC1CC(C(=O)N(CC(N)=O)CC(N)=O)N(C(=O)CCCn2cncn2)C1 C1(NC(COCCCCC)=O)CCN(C(c2cnn3c2CCCC3)=O)CC(O)C1 C1(C(=O)Nc2cccnc2)CC12CCN(C(c1cocn1)=O)C2 Cc1cc(CCCC(=O)NCCC2CCN(C(=O)C(C)N(C)C)C2)on1 c1(NC(CCN2CC(C(=O)OC)C(C3CCC3)C2)=O)ccc(F)c2c1CNC2 C1(CCC(=O)NCc2cc[nH]c2C(=O)NCCCN2CCC2)CCCOC1 CC(C)(C(=O)NC(C1CCCN1C(C12CSCC1C2)=O)(C)C)C(F)F C=CCCC(C(=O)NCCCCCCOC)NC(=O)CC(C)=C(C)C c1(C(N2CC(O)(C(C)NC(C3CC(CC)C3)=O)C2)=O)csc2c1CCCC2 Cc1cc(C)c(C(N2CC(NC(=O)C(c3ccccc3Cl)C)C(O)C2)=O)c(O)c1 c1(C(=O)NC(C(CO)NC(CC2CCN(CC)C2)=O)C)cccc(OC(F)F)c1 Cc1cnc(N2CCC(c3nncs3)C2)c(S(=O)(=O)NCCCCCC(C)C)c1 c1(C(N(C(C)CNC(=O)C(O)C=C)CC)=O)cccc(C)c1 c1(N2CC(CN(C)C(c3csnc3Cl)=O)OCC2)ncc([N+](=O)[O-])cc1C(N)=O CCCC(C(=O)N1CC2CC1C2CNC(=O)C=C(C)C)NC(=O)NC1CC1 c1(N(C)C(c2cc(S(C)(=O)=O)ccc2O)=O)nccc2c(Cl)cccc12 C(=O)(C(C(C)(C)O)NC(=O)C(C)SC)N(C1CC(C#N)C1)CC N1(CC(=O)NCC2C=CCN2C(C2CC2(F)F)=O)CCCC2(CC2)S1(=O)=O N1(C(C2C(C#N)C2)=O)CCC(O)(CCNC(c2ccc(OCC(F)F)cn2)=O)C1 c1(OC)ccc(C(N2CCN(C(=O)COC(C)(C)C(F)(F)F)C(C)C2)=O)c(C)c1 C1(C(=O)Nc2cccc(C(N)=O)c2)CC12CCN(C(=O)CC1CCNC1)CC2 C1(CCC)CN(C(=O)C(=O)NCc2coc(OC)n2)CC1Oc1ccccc1 N1(c2ncc(C)c(C)n2)CC2CCCN(C(c3ccccn3)=O)C2C1 Nc1c(C(N2CCCC(O)(CCNC(C3CC(CF)C3)=O)C2)=O)nc(O)nc1O N1(C(CCN(C(=O)C(n2nccc2C)C)CC#C)=O)CCC(F)(C(=O)OC)CC1 N1(C(C=Cc2c(C)ncs2)=O)CCCC(NC(C2CC2CC(C)C)=O)C1C C=C(Br)CN=c1ccn2ncc(S(=O)(=O)NC3CCCC3CC)c2[nH]1 c1(C(=O)NCCC2CN(C(C3C(OC)CC3)=O)C2)cc([N+](=O)[O-])ccc1N CC(C)(C)C(CNC(C1CCOC(=O)CC1)=O)C(=O)NC1CC=CCC1 CCC(C)(C)CC(=O)NCC(C)(C(C)C)NC(=O)Cc1ncc(Cl)s1 C(CCF)(C(=O)NCC1NC(=O)NC1=O)NC(c1c(C)snn1)=O c1(C(=O)NCC(C)(CNC(C2(CO)CCOC2)=O)OC)cc(C)c(C)c(C)c1 N1(C(CCc2onc(C)n2)=O)CC2CC1CN2C(C1CCC(=O)N1)=O c1(CC(=O)NC(CCCNC(C2CC(C)C2)=O)C)cccc([N+](=O)[O-])c1 c12ccnc(n1)N2.CC(C(C)(C)C)=CCO c1(C(=O)NC2CN(C(CCOC(C)=O)=O)CC(O)C2)[nH]c2ccccc2c1Cl c1(C(=O)NC2CC(NC(CC(C)n3cccc3)=O)CC2O)cc(S(N)(=O)=O)c[nH]1 C1(C(N2C(CNC(=O)CC(O)c3ccccc3)CCC2)=O)CCc2cncn2C1 C1(F)(CNC(C2(C)C=CCC2)=O)CCCN(C(C2CC3(C2)CC(O)C3)=O)C1 N1(C(C2N(CCC)CCCC2)=O)CCC(NC(=O)CC2(N(C)C)CCC2)C(F)C1 C1(NC(C2C=CCC2)=O)CCC2(CC1)CN(C(C13CCCC1C3(F)F)=O)CCO2 N1(C(COCCC)=O)CCC(C)N(C(=O)CC(O)C(C)CC)CC1 c1(C2CCN(C(=O)NC(c3nncn3C)CC)C2)ccccc1Cl N1(C(CC)=O)CC(NC(c2ccc(CC=CCN3CCOCC3)cc2)=O)C(F)C1 C1(C(=O)NCc2ccc(C(=O)NC(c3cscn3)C)s2)CN2CCC1C2 C1(C(N(C)CC2CN(C(c3cnc(Cl)[nH]3)=O)CCO2)=O)CC1C1CC(F)(F)C1 C12CCCC1NC2.C(=O)(C(F)(F)F)NC1C(NC(C)=O)C1 c1(C(=O)NCCCC(C)(C)NC(CC2CC(OC)C2)=O)cc(C)cc([N+](=O)[O-])c1N C1(NC(c2c(C)nco2)=O)CC(O)CN(C(=O)CCOCC2CC2)C1 c1(C=O)cccc(C(c2cc(CS)on2)C2CCC2)c1.C1(C2CCC2)CCCC1 c1(OCCC(=O)NC2(CC=C)CN(C(C3C=CCC3)=O)C2)ccccc1C N1(C(C(=O)NC2CC2)c2ccsn2)CCOC(C2CCC2)C1 Cc1cc(C(=O)NC2COCCC2NC(C2CC2C)=O)nn1-c1cccc(Cl)c1 CCC(CCCC(=O)N1CC(C)=CC(C)C1)NC(c1cn(C)ccc1=O)=O Cc1cc(C)cc(C=CC(=O)NC(C)C(C(C)C)NC(c2ncccc2F)=O)c1 C1(C(N(CCN(C)C(c2ncccc2N)=O)C)=O)CC2CCC(C1)S2(=O)=O c1(C(=O)NCc2nc(CNC(=O)CCC3CCC3)sc2)cnn2cc[nH]c(=O)c12 c1(C(=O)NCCCCCCN(C(C(CC#C)C2CC2)=O)C)cc([N+](=O)[O-])c(C)s1 C#CCC(C)C(=O)N1CC(N2CC(NC(=O)CCc3c(C)n[nH]c3C)CC2=O)C1 C1(N(C(C2N(CCC)CCC2)=O)C)CCC(CNC(c2ncccc2Cl)=O)CC1 c1(C(C)C(=O)NCC(C2CCN(C3CCCC3)C2)=O)c(F)cccc1F C12CC3CCC(C1)N3C(=O)C(O)Cc1cn2nn1.O=C1CN(CC2CC2)C(=O)N1 N1(C(c2c(CC)c[nH]c2)=O)CC(C(=O)NCCc2cccs2)CC(C)C1 CCC(C)(C(=O)NCCC1CCCCN1C(=O)COCc1ccncc1)C(F)F CONC(=O)C(=O)N1CC(=O)CC1C(=O)NCc1c(F)cncc1F C1(NC2CCCC(SC)C2)CCC2(CCNC2)CC1 S(=O)(=O)(c1cccc(Br)n1)N1CCC2(C(C(=O)Nc3cncc(Br)c3Cl)C2)C1 N1(C(C(C)C2CCC2)=O)CC(NC(c2ccncc2)=O)CC12CCC2 C(N=c1[nH]cnc2[nH]ccc12)C1C(NC(c2c(O)ccc(OC)c2)=O)CCC1 CCC(CCCC(=O)NC1(c2ncc[nH]2)CC1)NC(=O)C=CC1CCOC1 c1(C(N(CC(C)(C)CNC(=O)Cc2ccsc2)CC)=O)ccc2c(c1)ncn2C C1(CNC(=O)CCOCCCCNC(=O)CC2CC2C(F)(F)F)CCC(=O)O1 C1(CNC(=O)CCCCSC)CN(C)CCN1C(c1sc(C(=O)OC)c(N)c1)=O c1(CC(=O)NC2CCN(C(CNC(CC)=O)=O)C2)c(C)nc(CC)nc1C C(=O)(C(F)CC1CN(C(C2CCCOC2)=O)C1)NC(C(=O)OC)C1CC1 C(=O)(C1(C)CCn2c(C)nnc21)N(CCCCN(C(C(C=C)O)=O)C)C N1(Cc2ccc(OC)nc2)CCC2CN(C(c3cccnc3)=O)CC2C1 C1(C(=O)NCC(=O)NC2CCC2CNC(=O)CCCN2CCCC2)CCC(=O)N1 c1(-c2n(CCOC)c(N(CCS(C)(=O)=O)C)nn2)cnn2c1CCCC2C Cn1ccc(C(N2CC(O)(CNC(=O)CC3CSC3)C2)=O)c1 CC1CC(NC(=O)CCc2ccoc2)CN(C(C23CCCN2CCC3)=O)C1 C(c1ccco1)=C(C)C(=O)NCC(CNC(=O)C=CC(=O)N(C)C)CO n1(CC(=O)NCC(CC)NC(=O)C(C)OC)cc(C(=O)OC)cn1 N1(C(COC(C)C)=O)CC2(NC(=O)C(c3cc(F)cc(Cl)c3)=O)CCCC2(F)C1 c1(C(N(CCCCCNC(C2(COC)CC2)=O)C)=O)cnc(O)c2cccnc12 N1(C(C(CC)Sc2ccccc2)=O)CC2CC1(C(=O)N(CCCN=[N+]=[N-])CC)C2 C(=O)(C(CNC(=O)CCC1CC1C)CC(C)C)N(CCCO)CC c1(C(=O)NC(CN(C(C2C(C(=O)OC)C2)=O)C)C)cc2ccncc2[nH]1 CCCCC(CC)C(=O)N1CCCCC1CN(C(=O)COC)CC N1(C(ONC(C2CCCC2)=O)=O)CCCCC1Cn1ccnn1.C1(C)COC(=O)N1 CC12CCC(C(=O)NCC3(CNC(c4[nH]ccc4-c4ccccc4)=O)CC3)(C1)OC2 N1(C(C(CC)CO)=O)CCC2(CCC2)C(NC(c2cccc(COC)c2)=O)C1 CC(CN1CCOCC1)C(=O)NCCCC1(NC(=O)CN2CC3CC3C2)CC1 c1(CC)ccc(NC(=O)NC(CO)(CSC)NC(=O)NC)c(C)c1 C(=O)(CC(C)(C)COC)N(C1CCCN(C(=O)CCC2CC(OC)C2)C1)CC Cc1cn2nc(C(N3CCC(NC(c4coc(Br)n4)=O)C(F)C3)=O)cc2c(=O)[nH]1 CC(C)C(CCCC(=O)O)NC(C1C2CCC(C2)C1c1ccccc1)=O c1(OCC)nc(C)c(C(=O)NC2CCN(C(=O)CCC(C)OCC)C2C)s1 C(CC(=O)NC1CCC(CNC(c2c[nH]c3ncccc23)=O)C1)(C(F)(F)F)OC N1(C(C2C(C)=C2)=O)CCC(N(C(=O)CC2CC2)C)C1 c1(C(=O)NC(C(C)C)CO)ccc2c(c1)N(C)C(=O)CO2 C(N=c1cc[nH]c(-c2ccnn2C)n1)C1N(C)CCCC1(C)C N#Cc1nc(Cl)ccc1NC(C1CC(F)CN1C(=O)CCN1CCCCC1)=O C1(NC(c2cncs2)=O)CCN(C(=O)NOC2CCC2)O1 C(C(C)C(=O)NC(C(=O)N(CCCN(C)C)CC)=O)SC.C(C(F)(F)F)NC c1(C(N(CC(=O)NCC2CC(OCC)C2)CC(C)C)=O)ccc2cncn2c1 c1(OC)cccc(F)c1C(N1C(C(=O)Nc2cc(Cl)cc(Cl)n2)CC2CC12)=O C(=O)(C1Cc2ccccc21)N1CCN(C(=O)NCCC(S(N)(=O)=O)c2ccccc2)CC1 O=C1CC(C(=O)NCCC2CCCCN2C(=O)CNC(c2cnc[nH]2)=O)C(=O)N1 Cc1nc(C(N2CCC(C)C2C(N2CCCC2(C)C2CCC2)=O)=O)ccc1C#N N1(C(C2(C(CC)=O)CC2)=O)CCC1C(=O)N(C(C)C(C)C)C1CC1 C1(NC(C2(C3CCCC3)CCC2)=O)CC1C1CCCN(C(C2CCCCO2)=O)C1 c1(C(N(C(CN(C(c2[nH]cc(C)c2C)=O)C)C)C)=O)nnc(O)nc1O c1(C(N2CCCC2)CO)ccccc1Cl.c1(CC)noc(C)n1 CC(C)CC(C(=O)N1CC(C(C)NC(c2nn(C)cc2Br)=O)C1)C(C)C CC1OCCC1CC(=O)NCC(=O)NCC1CCCS1 c1(SC)ccc(O)c(C(=O)NC(C2CN(C(c3cc(Cl)cn3C)=O)C2)C)c1 Cc1cc(Cl)cc(C)c1OCC(N1C2CCC1CC(NC(=O)CCC(C)C)C2)=O c1(C(N(CC(=O)N(CC(C)O)CCN)C)=O)ccc2cnn(C)c2c1 N1(C(C(CCC)C)=O)CCC(NC(=O)CNC(c2cccc(F)c2)=O)C1(C)C Nc1cc(C(N2CCCCCC2CNC(=O)C=C2CCOCC2)=O)cc(Cl)n1 C(=O)(C(F)C(CC)CC)NC1(C(N(CCCC)C)=O)CSC1 c1(C(N2C(CO)CC(NC(c3cnc[nH]3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 c1(OC)nc(C)ncc1C(=O)NCC1CC(NC(c2cc(C(F)(F)F)on2)=O)C1 C1(CC)CCN(C(=O)C(NC(=O)C(C)n2ccnc2)SC)CCO1 c1(C(C(=O)NC2CC(NC(C=CC(=O)N(C)C)=O)C2)(C)C)ccc(Cl)c(Cl)c1 C1(NC(C(OC)OC)=O)CC2(CCC(CNC(C3CC(S(C)(=O)=O)C3)=O)CC2)C1 c1(NC2(CO)CCN(CC=CCCCCC)C2)nc(-c2ccccc2)ncc1C Cc1cnc(C)c(C(=O)NCC2CN(C(=O)CCOC3CCOCC3)CCO2)c1 C(=O)(CCC(CF)CF)N(C(C(=O)NCc1snc(C)n1)(C)C1CC1)C c1(CC(=O)NCCOCCN(C(c2cn(C(C)C)nn2)=O)C)cccc(C#N)c1 N#Cc1cccc(OC(c2cc(OCC=Cc3ccccc3)co2)=O)c1.C1CO1 c1(C(=O)NCC2C(C)CN(C(=O)CN3CCOCC3)C2)cc(C(N)=O)cc(F)c1 C#CC1CN(C(C2CCCCN2C(c2cccc(C)c2)=O)=O)CCO1 n1(CC(=O)N(C2C3CN(C(C(CCC)O)=O)CC32)C)ccc(O)nc1=O C1(NC(COCCC#C)=O)CC(CO)N(C(=O)C=CC(c2ccccc2)=O)C1 CC1CCCC(C)N(C(C2(C(=O)NC3CC34CCCCC4)CCCO2)=O)C1 c1(OC)ccc(CNc2ncccc2NC(C)CC#N)c(C)c1C C1(NC(C(C)(C)OCC)=O)CCC(C)(CNC(c2cc(C3(C)CC3)n[nH]2)=O)C1 C#CCC(CC(=O)NCC1CC2CCC1CC2)NC(C1CCCC(=O)C1)=O c1(OC)cc2c(cc1S(=O)(=O)N1CCN(Cc3nc(C(C)C)no3)CC1)CCC2 CN1N=CC(CC(=O)NCc2n[nH]cc2C(=O)NCCN(CC(F)F)C)C1=O Cc1cc(C#N)cc(C)c1C(=O)NCCOCCNC(=O)CCCCCF C(=O)(C1CCCc2ncc(C)n21)N1CC(CC=C)(NC(=O)C(C)CC2CC2)C1 c1(OC)ccc(C(=O)NC(CNC(c2csnc2C)=O)C2CC2)c(F)n1 N1(C(C(C)=CC2CC2)=O)CC(CNC(c2nccnc2N)=O)C2(CC2)C1 CC1(C)OCC2CC12C(=O)N(c1ccccc1Cl)C1CCCC1 Cc1nc(N)cnc1C(=O)NCC1CCCC(CNC(c2csc(O)n2)=O)C1 N1(C(C(C#N)=CC(C)C)=O)CCC(C)(C)C(CNC(C2CCOC(C)C2)=O)C1 C#CCC(CC#C)C(=O)N1C2CCC1CC(N(C)C(C1CC(F)C(=O)N1)=O)C2 N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NCC(O)CO)CC(C)C1 CC1(C#CC(=O)N2CC(O)CCC2C(=O)NCCCn2ccnc2)COC1 CC(C(=O)NCC1CCC1NC(=O)CCC1CC1)c1cc[nH]n1 c1(N2CCN(c3c([N+](=O)[O-])cccc3)CC2)ccc([N+](=O)[O-])cc1F N1(C(C(c2ccccc2)C)=O)CC(NCc2cc(Cl)n(C(C)(C)C)n2)C(F)C1 N1(C(C(c2ccc(OC)cc2)C)=O)CCC(NC(=O)C(C)=C(C)C)C(C)(C)C1 C1(CC)CCN(C(C2(N(C)C(c3cnc(Cl)s3)=O)CC2)=O)C1 c1(C(N2CCC(NC(CCC=C(C)C)=O)C2(C)C)=O)cc(O)cc(C#N)c1 C#CC(C1CCc2ccccc21)Oc1cccn(C(C)C)c1=O C1(CNC(C(C)OCC)=O)C2CN(Cc3ncnn3C)CC12 C1(CNC(c2c(C)cns2)=O)C2CN(C(c3c[nH]nc3C3CCCO3)=O)CC12 C12(C(=O)NCc3c(C)scn3)CC(CO1)N(C(=O)Cn1cc(C#N)cn1)C2 c1(OC)ncnc(OC)c1C(=O)NCCC1(C)CCN(C(c2cccs2)=O)C1 N1(C(C2CN(C(C)(C)C)C(=O)C2)=O)CC2CN(C(c3ccccc3C#N)=O)C2C1 c1(C(N(C2CN(C(Cc3c(OC)scc3)=O)C2)C)=O)cc(Br)n(C)c1 Cc1cccc(C(N2CC=CC(NC(=O)Cc3ccoc3C)C2)=O)c1N C(=O)(C(F)(F)C(F)F)N1C(C(=O)NC2CC(Cl)(Cl)C2)CC2CC21 n1(CC)cnc2[nH]c(=NC(C)c3cnsc3)nc(N3CCOCC(CC)C3)c12 O=C(C1=CCSC1)N1CC(O)(c2cn(-c3ccc(F)cc3)nn2)C1 C1(COC)CN(C(c2ccc(C)cc2F)=O)CCN1C(=O)Cc1ccc(OC)s1 c1(NC2(c3n(CC(=C)C)nnn3)CC(CCC)C2)cnc2ncccc2c1 c1(N(C)CC2CCN(C(C3CS(=O)(=O)C3)=O)C2)nc2c(cc1C#N)CCC2 C1(c2scc(CC(=O)NCC(C)(C)CO)n2)COCCN1C1CCCC1 N1(C(C(CC)=CCCC)=O)CCC(O)(C(C)NC(=O)C=CCN2CCCC2)C1 C1(NC(c2c(C)ccs2)=O)CC2(C1)CC2NC(=O)CCC(=O)C1CCN1C.C(C)(C)(C)S C1(CC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(C1CN(C(N)=O)C1)=O c1(C(N2CCC(C(=O)NC3CCNC3=O)(OC)C2)=O)nnc(O)nc1O C12(C(=O)NCC3CN(C(c4c(C)ncs4)=O)C3)CCC(CC1)C(C)(C)O2 c1(C(N2CC(C(=O)NC3CCCC3O)C3(CCC3)C2)=O)ccc2ncncc2c1 C1(O)(C(C)NC(=O)C2=CCSC2)CCN(C(c2cc(C3CCOC3)[nH]n2)=O)CC1 CCCC(CC)C(=O)N1CCN(C(c2cc(F)ccc2NC)=O)CC1C C#CCCN=C(NCC1CC2CCC1CC2)NC1CCCCC1(F)F c1(C(N2CC(CC)C(NC(=O)C(C)SC)C2)=O)cc(C)c2n[nH]cc2c1 C(=O)(C1=C(Cl)CCC1)NCC(CC)NC(=O)C(CN(C)C)c1ccccc1 Cc1[nH]nc(C(=O)N(CC(O)CN(C)C(=O)C2CC2C2CC2c2ccn(C)n2)C)c1C Cc1c(C(=O)NC2CCCC2CNC(=O)CC=CC(C)(C)C)sc2ccccc12 c1(OC)ccc(C(=O)NC2CCN(C(C34C=CC(CC3)C4)=O)C2)c(F)c1 N1(C(C(NOC)=O)=O)CC2(C=C(C(=O)NC(C)CCOC)CO2)C1 N1(C(c2cn(CCNC(c3ccoc3Cl)=O)nn2)=O)CCCC2(CCC2)C1 CCCC(CNC(=O)CC1COCCN1C(c1cccc(F)c1N)=O)CCC CC1(C)COCCC1C(=O)NC1CC(CC(=O)NCC2CSC2)C1(C)C C(=O)(CC(C)(C)CCC)NCC(CC=C)NC(c1cc2c(s1)CCSC2)=O C1(NC(c2cc(O)ccc2Cl)=O)CCN(C(c2cc(C3CC3)on2)=O)CC1F C(=O)(CCCCC(N)=O)NC(CN(C(C1CCCC(C(=O)OC)C1)=O)CC)C N1(c2nccc(C)n2)CCC2CN(Cc3cc(C(=O)O)cc(C)c3)CC2C1 C1(NC(c2cc(C3CC3)ns2)=O)CN(C(C2CC(OC(F)F)C2)=O)CC12CC2 C1(N(c2cnc(O)s2)Cc2ccc(F)cc2)CCC(c2cccc(F)c2)CC1 c1(C(=O)NC2CCN(C(c3ccnc4[nH]nnc34)=O)C2)cc2c(Cl)ccnc2s1 c1(C(=O)NCCC2(O)CN(C(c3cnc(C(C)(C)C)s3)=O)C2)ccc([N+](=O)[O-])o1 S(=O)(=O)(c1ccc(C(=O)NC2CCCC2NC(=O)COC2(C)CCCC2)o1)NC C(=O)(C(C)(O)C(F)(F)F)Nc1scc(CC(=O)Nc2cccc(OC)c2OC)n1 c1(C(N2CCN(C(C(=O)N(C)C)=O)C3C2CC3)=O)cc2c(=O)[nH]ccn2n1 N1(C(CC(=O)NCC)=O)CCC2(NC(=O)Cc3cc(F)ccc3O)CC2C1 C1(NC(c2cccc(C(=O)NC)n2)=O)CCCN(C(=O)C(F)n2ccnc2)CC1 C12(OC)CCC(C(=O)NC(C)(C)C(C)NC(C3C4CCCOC34)=O)(CC1)C(=O)C2 N1(C(c2cnc(COC)s2)=O)CCC2(C1)CN(C(C1CCOC1C)=O)CCO2 C1(CC(=O)NC2(CCC)CCNC2=O)CN(C(c2c[nH]nc2CC)=O)CCC1C N1(C(C(C)CC2CC2)=O)CCC(NC(c2cc(Cl)cc(Cl)c2)=O)C12CC2 C(=O)(CCCS(=O)(=O)N1CCCC1)N1CC(NC(C2(CCC=C)CC2)=O)C(C)(C)C1 C1(NC(c2nc(OC)nc(O)c2)=O)CCCC12CN(C(C1CC1C#N)=O)C2 C1(CNC(CC)=O)CC(F)(F)CN1C(=O)C(C)C(F)(F)F Cc1ccnc(C(=O)NCC2(C)CCCN(C(c3cccc(O)c3Cl)=O)C2)c1F n1(CC(=O)NC2(C)CCC2)ccc(C2CC2)n1 N1(C(C=CC)=O)CC(C)(C)OCC1CC.c1(N2C3(CC3)C2=O)ccc(C)c(C)c1 C1(C(N(CCCCC=C)CC=C)=O)COC2(CCC2)C1O CC1CCN(C(c2ns[nH]c2=O)=O)C1C(=O)NCCc1cocn1 CC(C)C(C)(CNC(c1cc(C2CCC2)no1)=O)NC(C1CC(F)(F)C1)=O C1(C(N2C(CNC(c3cc(C(F)F)cs3)=O)CC(O)C2)=O)CC2C=CC1C21CC1 c1(-c2scc(C(C)OC)n2)cccc(OCCOc2ccc(C)cc2)c1 C1(C(=O)NC2CN(C)C(=O)CC2)CN(C(C2(CN(C)C)CC2)=O)CC(C)(C)C1 c1(CC(=O)N(CC=CC(=O)NC(CCOC)(C)C)C)c(C)cnn1C C1(c2nnnn2C(C)C)(NCc2c(C)c(Cl)ccc2)CC2OC(C)(C)OC2C1 Cc1cccc(C(=O)NC2CCC(NC(c3cc(C(F)(F)F)nn3C)=O)C2)c1 C=CC1CN(C(c2cnc(OC)c(CC)c2)C(=O)NC2CCOC2)CC1O N1(C(C(C)Cc2ccccn2)=O)CC2CCN(C(c3csc(C#N)c3)=O)C2C1 C(CCC(C(=O)NC1CCCCCC1C)NC(c1ncncc1C)=O)OC c1(OCC(=O)NC2CCCC(NC(c3n(C)ccn3)=O)C2)cccc(Cl)c1Cl c1(NCCOC(c2ccc(C)cc2)CC)cccc(C2CCOC2)c1 Cc1ccc(CCNC(c2nnnn2C)(C2CCOC2)C)c(F)c1 C1(NC(c2c(N(C)C)ccnc2)=O)C2Cc3ccccc3C12.C1(C(=O)N)CN(C(N)=O)C1 Cc1nc(N2CCC(NC(=O)Cc3cnoc3)C2C)c2c[nH]nc2n1 CC1CCN(N2CCCC2c2ccccc2)CC1C(N)=O c1(C(N2CCC(C)C2c2cn(CCF)nn2)=O)cc(C(C)=O)ccc1C C1(C(=O)NCC(C2N(C(CSC)=O)CCC2)(C)C)CC2(C1)CC(CO)C2 C#CC1(O)CCCN(C(=O)CNC(=O)CN(C(=O)CCC2CCCOC2)CC)C1 c1(C(=O)NC(CCCNC(C(CC)SC)=O)C)cc2c(C)c(C)ccc2[nH]1 C1(C(N2CCCC(NC(c3n(CC)c(O)nc3)=O)C2)=O)COC(C)(C)CO1 Cc1cnc(C(c2nnnn2C)NCCCn2ccnc2C)nc1 N(C(=NCCCn1cncn1)N1CCC(Oc2ccccc2F)C1)C(C)C c1(NC(=O)NCC(COC(CC)(C)C)O)ccc(-n2cccc2)cc1C c1(NCC(O)CN2CCN(Cc3nc(C)[nH]n3)CC2)cn(C)c2cccc(C)c12 C(C(C)(C)C#CC(=O)NCC1CCCNC1=O)NC(C(C(C)C)OCC)=O C1(NCCNC(=O)Nc2c(C(=O)OC)oc(Br)c2)CC(C)CC(C)(C)C1 N1(C(C2CC(C3CCC3)C2)=O)CCN(C(=O)CCC2CC2(F)F)C(CC(F)F)C1 C1(C(=O)NCC2C(CNC(=O)Cc3cnoc3)C2)CCCCC1(F)F C1(CCC(=O)N)CCC(O)CC1.CC1(C)C(C(=O)NCCCCC2CC2)C1C(F)F c1(CCC(=O)NCCOCCN(C(=O)CC2CC=CCC2)C)ccc(Cl)cc1 N1(C(CC2C(C(=O)O)CCCC2)=O)CC2C=CCC(C2)C1.c12cn(nn1)CC2 C(=O)(C1=Cc2ccccc2C1)NC1(CNC(=O)Cn2c(O)nnc2O)CC1 S(=O)(=O)(c1scc(Br)c1Br)N1C(c2n(C)cnc2)CCC1 c1(C(=O)OC)ccc(C(=O)NCC(CSC)OC(c2cn(C)nc2C)C)nc1 c1(C(=O)NC(CC(=O)NC(CC)CSC)(C)C)cc(O)cc(F)c1 c1(C(N2CCN(C(C(C)OCC=C)=O)CC2CCOC)=O)c(C)ccc(Cl)c1F C1(C(=O)NCC(C)(CO)NC(CC(CC)C)=O)CCN(OC)CC1 C(C(=O)NCC1CCN1C(c1cc(C)c(Br)o1)=O)(C(C)(C)C)OC C1(C)(C(N2CCC(O)(C(C)NC(c3ccc(-c4cccs4)[nH]3)=O)C2)=O)CC(C#N)C1 N1(C(c2cc(C)ncn2)=O)CCC2CN(C(=O)Cn3cc(C4CCC4)nn3)CC12 N1(C(CC2(C=C)CC2)=O)CCC(F)(CNC(=O)C(F)(F)c2cccnc2)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC(CC)C1CC1)N(CCOCC)CC C=CCN=c1[nH]cc(C(N2CCC(CNC(c3ccc(Cl)cn3)=O)C(C)C2)=O)s1 N1(C(C2N(CC)CC2)=O)CCC(CNC(=O)Cc2csc(C)c2)C(CO)C1 c1(CC(C(=O)NCC(N)C2CC2)NC(=O)OC)ccc(Br)cc1 O=C(NN1CCCC1C(N1CCC2CC1C(=O)O2)=O)c1ncc(F)cn1 Cc1cc(C(N2CC(CNC(c3cnn4c3CCC4)=O)C3CC23)=O)c(Cl)cc1F C1(CNC(Cc2cccc(C(C)C)c2)=O)CN(C(=O)CC2CSC2)CCC1C C(CCC(=O)NC(CNC(C1(OCC)CCC1)=O)CO)O.C1(=O)N(C)O1.C1(CC)CC1 C#CCCC(C(=O)N(C(CF)CF)C)NC(=O)CCOCC1CCCO1 CN1CCOC2(CN(C(c3cnc(Cl)s3)C(=O)NCSc3ccccc3)C2)C1 c1(C(=O)NC(CNC(CCCCC#C)=O)(C)CC)cc2cc(F)ccc2[nH]c1=O c1(OC)ccc(Cl)c(C(N2CC(O)(CCNC(=O)C(C)CN(C)C)C2)=O)c1N C(=O)(CS(=O)(=O)CCO)N(C1CCCCN(C(CC(n2ccc(C)n2)C)=O)C1)C C12(N(Cc3cncs3)Cc3c(CC)non3)CCCC1N(C(=O)CCS(C)=O)CC2 C12(C(=O)NC3(CC=C)CCN(C(C4C5CC(=O)CC45)=O)C3)CCN(CC1)CC2 N1(C(CCC2CC(NC)C2)=O)CC(CC(=O)N(CCC(O)CO)C)CC1(C)C c1(CN2C(C(=O)Nc3cc(C(C)=O)c(F)cc3)CSCC2)cc2ncccc2[nH]1 Cc1cc(C)c(C(=O)NC(C)C(C(C)C)NC(c2[nH]nnc2C)=O)o1 C1(NC(C2(OC)CCSC2)=O)CC(NC(=O)C(C2CCCC2)OC)C(O)C1 c1(C(=O)NCCN(C(=O)COC2CCC(C)CC2)CC)ccc2cnccc2n1 CCC(F)(F)C(=O)NC1CC1CNC(=O)CCCOc1ccccc1Br C1(CC(=O)NC2CCC(C(N(C(c3ccccn3)C)C3CC3)=O)C2)COCCOC1 Cc1cccc(C(O)C(=O)NC(C2CCN(C(C3(C4CC4)CC3)=O)CC2)C)c1F N1(C(C2C(C(C)O)C2)=O)CC(NC(c2[nH]nnc2C)=O)CC1C N1(CC(N2C(CNC(C(C)n3cccc3)=O)C=CC2)=O)CCC(C)(C)C1 C1(NC(c2c(CC)occ2)=O)CCCCC12CCN(C(C1CCSCC1)=O)C2 CCCC(O)(CCC)CC(=O)NC1CN(C(c2oc(SC)cc2C)=O)CC1SC Cc1ncnc(C)c1C(=O)N(CC(C)(C)NC(C1CS(=O)C1)=O)C c1(C(=O)NC2C(C)N(C(=O)CCC(C)(C)C)CCC2C)ccc2c(c1)CC(=O)N2 C(c1cc(Cl)sc1Cl)=Cc1nnc(CCCC)o1 C#CCCCCCC(=O)NC1CC(C)CN(C(C2CCCN2C(N)=O)=O)C1 CCC(C)(CC)C(=O)NCCC1CCCN(C(=O)C(C)Sc2ccccn2)C1 c1(N2CCC(NC(C3CC(C#C)(O)C3)=O)C(C)(C)C2)ncnn2c(Br)ccc12 C(=O)(CC1OCCc2sccc21)NCC(C(C)(C)C)N.N1(S(=O)(=O)CC)CCCCCC1 N1(C(C(C(C)C)NC(CC(=O)NCC)=O)=O)CCC2(CCC2)CC1 C1(O)(C(=O)NC2CCC(CNC(C(C(=O)OC)C)=O)C2)CCCCCC1 c1(N(CCCN(S(C)(=O)=O)C)C(=O)NC2CC23CC3)ccccc1 c1(C(=O)NCC(CC=C)NC(c2c(C)n[nH]c2C)=O)cc(C)ccc1[N+](=O)[O-] CCC(C)(CNC(=O)C(C)(C)CCNC(c1cn(C(C)C)cn1)=O)C(C)O C(=O)(C(F)(F)C(O)C(C)C)N(c1nnn(CC)c1N)CCCC(C)COC(C)=O S(=O)(=O)(c1cnc(N(CC(C)C(F)(F)F)C)c(Cl)c1)NC(C(CC)C)CO N1(C(COCCOCC)=O)CC(NC(=O)C(c2ccc(F)c(Cl)c2)C)CC(F)C1 c1(C(N)=O)ccccc1C(=O)NCC1CN(Cc2ccncc2Cl)CCO1 C(=O)(C1=C(C2CC2C)N(C)C(=S)NC1c1ccc(O)c(OC)c1)OC c1(C(C(N2CC(O)(CNC(C3CN(C(C)C)C3)=O)C2)=O)O)cccc(Br)c1 CCCC(C)(C)CC(=O)N1CCOC(CNC(c2cc(Br)ncc2O)=O)C1 c1(C(=O)NCC(C2CCC2)CNC(c2n(C(CC)C)ncc2)=O)cc(O)nn1C O=C(CC1=NNC(=O)C1)NCC1CC(CNC(c2cncc3c[nH]nc23)=O)CO1 c1(C(N(C(C(=O)NC(CC(=O)OC)C)C)C2CC2)=O)cncc(OC)c1 c1(C(C)N(C(CC2CCCC2)C(=O)NCC2CCOC2)C2CC2)cccc(Br)c1 C1(COC)(CNC(=O)CC2(O)CCCC2)CN(C(=O)CSc2nncn2C)C1 C1(NC(c2cc(C)[nH]c2)=O)CC2CC(NC(C3CC4CC4C3)=O)C1C2 c1(C(=O)NCC2(O)CN(C(c3c(CC)n(CC)nc3)=O)C2)ncc(F)cc1F C1(C(N2CC(CC(C)NC(CNC(C)=O)=O)C2)=O)CC2(C1)NC(=O)NC2=O C1(NC(CCCCCC=C)=O)CCC2CCN(C(=O)CCCC)C1C2 C1(NC(C(C)C)=O)CC2CN(C(=O)C(c3cc(F)cc(F)c3)C)CC2C1 C1(NC(=O)NC(C)C=CC(=O)NC2CN(C3CCC3)C2)CC2(CCC2)C1 C1(CC(=O)NCC2(CN(C(c3c(C)nco3)=O)C)CC2)CC(C)CC(C)(C)C1 C1(NC(COC(CC)(C)C)=O)CS(=O)(=O)CC1NC(=O)C(F)(F)C1CC1 c1(N(C)CC2CCN(C(Cn3nc(C)oc3=O)=O)C2)ncc([N+](=O)[O-])cc1C Cc1cc(S(=O)(=O)N2CCC(n3cccn3)CC2)c(C)cc1[N+](=O)[O-] C=C1COCCN(C(c2nn(C)c(Cl)c2C(F)(F)F)=O)C1 C1(C)(NC(C=CCOCCOC)=O)CCN(C(=O)CC(CC)C2CC2)C1 C1(NC(C(CCC)C)=O)CC2CC1N(C(=O)CCCc1nc(C(C)C)no1)C2 c1(OCCCOC)ccc(-c2ccc(NC(=O)C(C)CSC)cn2)cc1 c1(C(C(=O)NCC)N(CCN(C)C)Cc2ccc(C)s2)onc(Br)c1C CC1(CNC(C2CCC3CC23)=O)COCCN(C(c2cccc(Cl)c2F)=O)C1 c1(-n2c(-c3c(Cl)cccn3)nc(Cc3cccnc3)n2)nc2ncccn2n1 N#Cc1c[nH]c(C(=O)NCC2(NC(C34CC(CO3)C4)=O)CCC2)cc1=O C1(F)(CNC(c2c(CC)ncs2)=O)CCN(C(C2CCC23CCCO3)=O)CC1 c1(-c2cn(C(C(=O)OCC)C)nn2)ccc2[nH]ccc2c1 C12(CNC(=O)Nc3ccc(Cn4cccn4)o3)COCCN1C(=O)COC2 C1(CCOC)(NC(C2COC(C)C2)=O)CCN(C(=O)C=C(C)C2CC2)CC1 C(C(C(=O)N(CCO)CC)NC(C1CCNC1=O)=O)OCC Cn1ncc2c(C(=O)NC3CC(F)(CNC(=O)Cc4cnsc4)C3)ccnc12 C(=O)(CC1=NN(C)C(=O)C1)NCC(CC(C)C)NC(=O)CCOC1CCOC1 C1(C(=O)NC(C(=O)NCC(=O)N(C)C)C2CCCO2)CC2(CCCO2)C1 C1(C(=O)NCC(c2c(OC)cccc2)NC(C)=O)COCCC1(F)F C(=O)(C(O)CC[S+](C)C)N(C(C)CNC(c1cn(Cc2ccccc2)nn1)=O)C C1(NC(C(C(=C)C)(C)C)=O)CN(C(=O)COCC(=O)NC)C2(CCCOC2)C1 C(C(=O)N1CC(O)(CNC(=O)Cc2cnns2)C1)(C(F)(F)F)OC(C)=O C1(NC(c2cnc(C)o2)=O)CCC(CC(=O)NCCC2CCCCO2)CC1 Cc1cc(C(N2CC3(CC(NC(C4(C)CNC(=O)C4)=O)C3)C2)=O)c(F)cc1Cl c1(C(=O)NCC(CC(C)C)NC(c2c(CCC)n(C)nn2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nccc(C(=O)NCCCN(C(=O)C(O)C(C)C)CCO)c1N C(C)(CC(C)C(F)F)NC(C1(F)CN(C(c2ccc(OC)cn2)=O)C1)=O C(=O)(CS(=O)(=O)NCC)NCC(CC=C)NC(=O)C=Cc1cc[nH]n1 c1(OC)ccnc(C(N2CCC(N(C(=O)C(C)(C)SC)C)C2)=O)c1 Cc1cc2[nH]c(C(N3CC(C4CN(C(=O)Cn5[nH]cnc5=N)C4)C3)=O)cc2o1 c1(C(=O)NCC2=CCN(C(CCOC)=O)CC2)cccc2c1OC(C)C2 C(CCC(C)C(=O)NC(C)(C)CNC(c1cnc(C)c(C(F)(F)F)c1)=O)OC N1(C(C2(CC)CN(C(=O)CS(C)(=O)=O)C2)=O)Cc2ccnn2CC1C C1(NC(C(N2CCC(C)CC2)=O)=O)CN(C(=O)C(C)(C)CC2CC2)CC2(CC2)C1 Cc1ccc2c(c1)SC(C(N1CC3(CCC(NC(C4(CF)CC4)=O)CC3)C1)=O)C2 c1(CC)cc(F)ccc1C(=O)N(C)CCNC(C1CNC(=O)C1)=O c1(C(=O)NCC(C2CC2)NC(c2ncsc2C2CC2)=O)cnn2c1CCC2 c1(C(=O)NCC23CC2CN(C(C2CCC(C(F)F)CC2)=O)C3)cc([N+](=O)[O-])cs1 Cc1[nH]nc(Cl)c1C(N1CCCC1CNC(=O)CC1CC1)=O CCCC(CC)C(=O)OC(c1ccc(F)nc1)C C1(CCNC(C2CC2c2cccs2)=O)(OC)CN(C(=O)C(F)(F)C2CC2)C1 C(=O)(C(C)CC(C)C)NC1C(CC(=O)N(CC=C)CCOC)CCCC1 C1(C(=O)NC2CN(CC)C(=O)C2)CCCCCCN1C(c1occc1C)=O c1(C(=O)Nc2cc(-c3cc(N)c(F)cc3)cc(F)c2)cccc2nc(O)ccc12 N1(C(CS(=O)(=O)NCC)=O)CC2CC(C(=O)NCC3(CSC)CCC3)C(C2)C1 Cn1c(C(=O)NCC2(C)CCC(NC(c3cc(C(C)(C)C)c[nH]3)=O)C2)cnc1S N1(C(c2c(C)nc(CCC)s2)=O)CCCN(C(=O)COCCOCC)C(CO)C1 n1(CC(=O)NC(CC)CNC(=O)Cn2nc(C)nc2C)c(C)cc2ccccc12 C1(CC(=O)NCc2c(C(=O)NCC=CC)occ2)CCC(C)CO1 C1(NC(CCCc2cc(C)sc2C)=O)CCCC(NC(c2cnccn2)=O)CC1 c1(C(=O)NCCC(C)NC(CCCCSC)=O)ccccc1S(=O)(=O)N(C)C C1(N(C(C(OC)OC)=O)C)CCC(NC(c2n[nH]cc2C2CC2)=O)CC1 N1(C(C(N2CCC(C)(OCC=C)C2)=O)=O)CC(C)CCCC1C N1(C(c2nc(C)oc2)=O)CCOCC1CNC(C1CC(=C2CC2)C1)=O C1(CN(C)C)(NC(c2[nH]nc(Br)c2Cl)=O)CCOCC1 CC1CCc2ncc(C(=O)NCC3(NC(C4CCCCC4)=O)CCCCC3)n2C1 C1(C(=O)NCCC(C(=O)NC2CCNC2=O)OCC)CCCCC1(C)C N1(CC2C(C)CCC2)C(=O)CCN(CCc2cccc(Cl)c2)C1=O CC1C(NC(=O)C=Cc2ccncn2)CCN1C(=O)CNc1ncccn1 CCCCC(O)C(=O)N1CCC(C(C)NC2(C(=O)OCC)CCCC2)C1 c1(SCC(=O)NCCN(CCOC)C(C23CCCC2C3)=O)cccc(OC)c1 Cc1cc(C(=O)NC(CNC(c2snnc2C2CC2)=O)C2CC2)cc2ccoc12 CCC(C(=O)NCC1CCC(NC(=O)CCC=C(C)C)C1)C(F)(F)F c1(CC(=O)N(C2CCCC2)CCNC(c2cnc(CSC)o2)=O)ccncc1Cl C1(NC(=O)NC2CC(C)(CC)NC2=O)CCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 N1(C(CCN(CCCCC)C)=O)C2CCC1C(COC)NC2 N1(C(C(CCCC)F)=O)CCC2CN(C(C3CCc4ncnn4C3)=O)C(C)C12 N1(C(C(C(=O)OC)C)=O)CCC(CNC(C2CN(C(C)=O)C2)=O)C(F)(F)C1 c1(N(C(C2(CC=C)CN(C(=O)COC)C2)=O)C)ccc(CC)c(F)c1 C1(C(=O)NC2CCC(C)(C)C2)(NC(CCc2ccc(C)o2)=O)CCCCC1 CC1OCCC1(F)C(=O)NCCN(C(c1coc(O)n1)=O)CC1CC1 C(C(=O)NNC(=O)CNCc1ccc(C#N)c(Cl)c1)c1ncn(C)c1 c1(CC(=O)NC2C(NC(c3c(C)cn(C)n3)=O)CC2)ccc2n[nH]cc2c1 n1(C(C(=O)NC(C(=O)OC)C2CCCC2)C)cc(CCOC(=N)O)nn1 Cc1noc2cc(NCCNC(c3ccc([N+](=O)[O-])cc3)=O)ccc12 C1(NC(C(N(CCCOC)CC=C(C)Cl)C2CC2)=O)CCOCC1 C1(NC(C(C)=CC)=O)CC2CCC1C(NC(c1cccnc1N1CCCC1)=O)C2 Cc1nsc(N2CCCC(NC(C3CCCC(=O)N3)=O)C2)c1C#N c1(NC(=O)CCCC2CCOCC2)cccc(NC(c2occc2Br)=O)c1 CC1(C)CN(C(C2(CC(F)F)CC2)=O)CCC1NC(=O)CN1CSCC1=O N1(C(C2N(C(c3cc(CSCC)on3)=O)CCC2C)=O)CCCOCC1C c1(-n2ncc(NC(C(C)NC(=O)NC3CC3)=O)c2)ccc(F)c(Cl)c1 C1(NC(=O)NC(c2ncccn2)(C)C)CCN(c2ccccn2)C1 C(CCCCCC(=O)NCC1CCOCC1)NC(c1c(C)c(F)cnc1)=O c1(C(=O)NCCCCNC(c2cccc(C(F)F)c2)=O)c(O)cc(O)cc1O C(C1CN(C(=O)CCc2cncnc2)CC1C(N1CC(C)C(C)C1C)=O)=CC c1(C(N(C(C)CCNC(c2nc(Cl)c(Cl)s2)=O)C)=O)cc(N)cc(F)c1 C1(N(C)C)CN(C(=O)Cc2ccns2)CC1CN(C(=O)C(O)CC1CC1)C1CC1 C1(C2CCN(C(C3(N(C)C)CC3)=O)C2)(NC(Cn2c(C(C)C)ncc2)=O)CC1 c1(OC)ccccc1C(C)CC(=O)NCc1nc(C(C)C)no1 C1(NC(c2cccc(C)c2)=O)CC2CC1CN(C(=O)COc1ccsn1)C2 C1(CCNC(c2n(CCCSC)nnn2)c2cnn(C(F)F)c2)CCC(C)(C)O1 CCCC(C)(O)CNC(=O)C(C1CC1)N(C)C(c1cc(CC)ccn1)=O c1(C(=O)NC2CCCN(C(CC(C)C3CC3)=O)CC2)cccc2[nH]c(=N)oc12 c1(C(=O)NC2CC2)cccc(C2(C(F)(F)F)CCC2)n1.c1(C(C)O)ccnn1C c1(C(N2C(C)(C)C(NC(=O)CNC=O)CC2)=O)cnc(O)c2cccnc12 c1(NC(c2n(CC)nnn2)c2cscc2C)ccc(Cl)c(C)c1 CCC(C)CCCC(=O)NC1CC2(C1)CN(C(C1CCC1c1nncn1C)=O)C2 C1(C(=O)NC(CC)CNC(C2CC2C2CCCO2)=O)CC(=O)NC(=O)C1 C1(C(=O)NC(C)CCSC)(OC)CCN(C(c2nccnc2N)=O)C1 c1(OC)ccc(C(=O)N(C2CN(C(C3(C)CC=CCC3)=O)C2)C)nc1OC n1(CC(=O)N(C(CO)C(C)C)C)nnc2c1C1C(=O)N(C1)C2.CN c1(C(=O)NCCC(C)NC(=O)Cc2cnccc2C(F)(F)F)snc(O)c1Cl C1(CC(=O)N(CCC(=O)NCC2CSCCO2)CC)CCCN(C)C1 c1(CC(=O)NC(=O)NC2CCN(CC3CCCCC3)C2)cccc(Br)c1 N1(C(c2c(SCC)cccc2)=O)C2CCC1C(NC(C1CC1(C)C)=O)C2 C(C(=O)N1CCC1CNC(=O)Cn1nnnc1C1CC1)(C(C)C)N(CC)CC N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCCC(N=c2nc(SC)[nH]s2)CC1 C(C(C)(CC)C(=O)NCC(C)(C)C#N)NC(c1n(C=C)ncc1)=O N(C)(C1CCc2ccccc21)CC(=O)N(c1n[nH]cc1C)CCCC N1(CC(CC)C)CCCC(F)(COC)C1 c1(C(=O)NC2CCN(C(C(C)(C(C)C)NC(C)=O)=O)CC2)cnc2scnc2c1 N1(C(c2cnc(CC)o2)=O)CC(C)CCC1CNC(c1cnnn1C)=O c1(OC)ccc(C(=O)NC(C)(C)CNC(C2SC3C=CC2CC3)=O)cc1C c1(COC)cc(C(=O)N(C2C=CC2C(=O)OCCC(=O)NC)C2CC2)n[nH]1 C12(CNC(C(CC)COC)=O)CN(C(C3SCCS3)=O)CC1CCO2 N1(C(c2c(C(C)C)noc2)=O)CCC(C)(CNC(=O)CC2CCOC2)C1 C(=O)(C1=C(Cl)CCC(C)C1)NCC1CCCC(NC(COCCCCC)=O)C1 CC1(C)CCC(F)(CNC(=O)NC2CCCO2)CC1 C1(NC(c2c(C)cc(C(F)(F)F)cc2)=O)CN(C(=O)C(C)O)CC2(CC2)C1 N1(C(c2ccc(OC)o2)=O)CCC(C)(C(=O)NCC2CC23CCC3)CC1 c1(C(N(C2CCCC(N(C)C(c3cnccc3Cl)=O)C2)C)=O)ccnc(S)c1 c1(C(N(C2CCCN(C(c3cnc(C(C)C)[nH]3)=O)C2)CC)=O)cc(N)c(F)cn1 C(=O)(C1CCCn2nccc21)NC1CCN(C(CSc2nc(C)[nH]n2)=O)C12CC2 C=C(C)CC(C(=O)OC)NC(C1CC(F)(CNC(=O)CCNC(C)=O)C1)=O CCCC(CC)C(=O)N1CC=C(CNC(=O)CN2CCOCC2)CC1 C1(NC(C(N2CCOC2=O)C)=O)CN(C(c2cnc(C3CC3)[nH]2)=O)C2(CCC2)C1 CCN(OC)C(=O)CNC(C1(C)C=CCN1C(=O)CN(C)C(C)=O)=O c1(CN2CCCC(NC(c3ccccc3I)=O)C2)ccc(Br)cc1C(F)(F)F c1(CC(=O)NC(CNC(CCc2ccc(C(=O)OC)[nH]2)=O)C)cnc(C)nc1O C1(CCC(=O)N(C(CC)COC)C)CCCCN(C(=O)C(CC)CCOC)C1 C(CN=c1ccc(C)c[nH]1)NCCCC1(CC(=O)OCC)COCCO1 c1(C(N2CC(C(C(=O)NCC3C=CCS3)O)C2)=O)cc2cccnn2c1 Nc1c(C(N2CCCc3ncccc32)=O)ncc2ccccc12 C1(CNC(c2cc(CNC(C3(NC(N)=O)CC3)=O)on2)=O)CCCOCC1 c1(C(=O)N)n[nH]c(C)c1Br.c1(CC)cccnc1NC(c1nnnn1C)C1CC1CO N1(C(C2N(C)C(=O)CC2)=O)CC2CC(C1)CN(C(=O)CC1(C#N)CCCCC1)C2 CCCCCC(C)CC(=O)N1CCC(CCNC(c2c(C)ccc(Cl)c2N)=O)C1 C12(CCN(C(=O)C(C)SC)C1)C(=O)N(C)C2.C1(C)(CC)CC1 C(CN=c1nc(N2CCCC(CC3CC3)C2)c2c([nH]1)COC2)(C(F)(F)F)OC C1(C)(C(N2CCC(OC)C2)=O)CCN(C(=O)C=CC2CCOCC2)CC1 c1(C(=O)NCCN(C)C(C2(C)CC2c2ccccc2)=O)coc2cccc(O)c12 N1(C(C2(C)N(C(C(C)n3ccnc3)=O)CC=C2)=O)CC2CCCCC12C c1(OC)ccncc1SN1Cc2nccc3c2OC(C)(C)C13 c1(C(N2CC(CC=C)(C(=O)NCC3CC4CCC4C3)C2)=O)cc(O)cc(F)c1 C(=O)(CC(C)(C)COC)NC(CNC(c1[nH]cc(CC)c1)=O)C1CCC1 C(=O)(C(O)CCc1ccco1)NCCC(=O)NO.C12CCN(CC1)NC2=O c1(C(N2CC(CC(=O)OC(C)(C)C)C2)=O)cc(-c2cccs2)[nH]n1 N1(N2CCCCC2)CCS(=O)(=O)CC1.C1(C(N2CCC2)=O)CCC(C2CC2)N1 C1(C)CCCC1.C(CCNC(C1CC1F)=O)NC(C1CC1F)=O c1(OC)cc(C(=O)NC(C)CN(C)C(C2CCOC2C2CC2)=O)cc(N)c1OC C12(C(N3CC(CCNC(c4scnc4C4CC4)=O)C3)=O)CCC(=O)N1CCS2 C1(C)(OCC)CN(C(=O)CNC(c2cncnc2)=O)C1.C12(CCC1)C(=O)N2 N1(C(C(C)NC(=O)OC)=O)CCCC(C)(CNC(=O)COC2CCCCC2)C1 C1(C(N2CCN(C(=O)OCC)CC2)=O)COCCN(C(C23CC(NC)(C2)C3)=O)C1 c1(OC)ccc([N+](=O)[O-])cc1CNC(C1(C)CCCN1S(=O)(=O)CC#N)=O c1(OCCCC)ccc(NC(=O)CN(C(C)CNC(=O)C(C)(C)C)C2CC2)cc1 N1(CC(=O)NCC(=C)CCNC(=O)CSc2ccccn2)CCCCC1=O N1(C(C2C(C=C)CC2)=O)CCC(C(C)(C)C)(CNC(=O)C=Cc2cnc[nH]2)C1 C(=O)(CCCCCNC(C)=O)NC1CC(F)(CNC(c2ccc(CC)[nH]2)=O)C1 C1(NC(c2c(CC)ccs2)=O)CN(C(=O)C=Cc2c(C)coc2C)CCC1F c1(Nc2cc(C(=O)O)c(Cl)cc2)ccn2c(C(=O)O)cnc2c1 C1(C(=O)NC(C=C)C(F)(F)F)CN(C(=O)C(C)O)CCC1(C)C c1(C(=O)OCC)cccc(N2CCOCC2)c1.C12CCC(C1)NCC2 Cc1ccc(C(=O)N(C2CCCN(C(=O)C#CC3CC3)C2)C)c(C)n1 C(=O)(C(C)P(C)(C)=O)NCCCCN(CCCS)C.N1(C(CSCC(C)C)=O)CCOCC1 C(CC(C)C)(C(=O)NC(C)CS(C)=O)N(C(CNC(CCC)=O)=O)C C1(C(=O)NC2CC(CNC(CC3CC(OCC)C3)=O)C2)CS(=O)(=O)CC(=O)N1 C1(C(=O)NC2(CCOC)CC2)CC12CCOC2.C1(C)C(=O)N1CC=C C1(C(=O)NCCCNC(=O)C(F)(F)CC2CC2)CCCC12CCOCC2 c1(C(=O)NCC2(C(N3CC4CCC3CC4)=O)CC2)cc(O)nc(O)n1 CCC(C)CC(=O)N1CC2CC2(C(=O)NCc2ccc(OC)cn2)C1 N1(C(C2=C(C)OCCS2)=O)CCC2CCCN(C(=O)C=Cc3ncc[nH]3)C2C1 Cc1cc(=NCCOCCO)[nH]c(NC2COCC2C2CC2)n1 Cn1cc(Cl)c(C(N2CCOC(C(=O)NCC3CNC(=O)C3)C2)=O)n1 C1(CC(=O)NC2(C(C3(C)N(C(C4C(C)C4)=O)CC3)=O)CCC2)CCC(=O)NC1.N C(CC(=O)NNc1nc(C(C)(C)C)cs1)c1nc(C#N)cc(C)n1 N1(C(CCCCC)=O)CC2(CCC2NC(c2ccc(Cl)c(F)c2)=O)C1 CCCCC(O)C(=O)NCC12CC(CC)(CN1C(c1c(C)ccnc1O)=O)C2 c1(NC(c2ccc(NC(CC(C)SC)=O)nc2)=O)cnn2ccccc12 N1(CC(N2C(C(=O)NCc3ccn(CC)n3)C=CC2)=O)C(=O)CNC1=O C1(CC(N2CCN(C(c3ccc(F)c(Cl)n3)=O)CC2)=O)CCC(F)(F)CO1 N1(C(C(C(C)C)C)=O)CCN(C(=O)CCC2CC2)CC1C C1(C(=O)OC)(C(=O)NC2CCC(N(C)C(c3cnsn3)=O)CC2)CCOCC1 c1(C(N2CCC(N(CCC)C(c3c[nH]nc3C3CCC3)=O)C2)=O)nnccc1C c1(-c2scc(C(F)(F)F)c2)ccnc(N2CCN(Cc3cscn3)CC2)c1 N1(C(C(C2CN(C(C3C(C)CCOC3)=O)C2)O)=O)CCC(F)(F)CC1 c1(C(N(CCN(C(C(C)C2CCC2)=O)C)C)=O)cccc(C2CCC23CCC3)c1 N1(C(c2c(C)cccc2)=O)CCC(O)(CN(C)C(C2CC3(C2)CC3F)=O)CC1 N1(C(c2cccc(C)c2)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC12CC2 c1(C(N2CCC(=CCNC(CNS(NC)(=O)=O)=O)CC2)=O)cc2sccc2n1C N1(C(C(CC)F)=O)C(CNC(=O)CNc2nccs2)CC2CC12 Cc1cc(C(N2CC(CNC(C3(c4ccc(Cl)c(F)c4)CC3)=O)C2)=O)ccc1Cl Cc1[nH]c2ccccc2c1C(=O)NCC1CC1CNC(C12CC(C)(CO1)C2)=O CC1=CC(O)CN(C(C2CNCC23CCC3)=O)C1 Cc1cc(C)n(CC(=O)NC2CC(CCNC(C3CCCCS3)=O)C2)n1 C(=O)(C#CC1CCOC1)NC1(NC(C2CCC(C(C)C)CC2)=O)CCC(C)(C)C1 c1(OC)c(C(=O)N(C2CCCN(C(=O)CCC3CC(C)(C)CO3)C2)C)csc1C CCC(C)C(C(=O)NCc1cc(C(=O)N(CCCO)C2CC2)n(C)n1)OC N1(C(c2nccc(C)c2N)=O)C2CCC1CC(CNC(c1ccnc(F)c1)=O)C2 c1(C(=O)NCC(C)CNC(=O)C(O)C2CC2)c[nH]cc1C(=O)NC1CCOCC1 C(=O)(C1CCCc2c1ncn2C)NCC(CNC(Cn1c(C)ccn1)=O)CO O=C(CC(CC1CC1)NC(C1CCC2(CC2)C1)=O)NC(c1ccco1)CO C#Cc1ccc(F)c(C(N2CC(OC)CC2CNC(=O)CC(C)CCC)=O)c1 c1(C(N(CCC(C)NC(=O)CC2CC(=O)NC2=O)C)=O)csc2nccn12 C(C(CC1CC1)C(=O)NC(C)Cc1ccco1)NC(CSCCCC)=O c1(C(N2CCCC(CNC(c3cc(Cl)ccn3)=O)C2)=O)cnc(O)nc1O C1(C(N2C(CNC(=O)CC3(O)CCC3)CCC2)=O)Cc2ccc(F)cc2C(=O)O1 c1(C(N2CCCC(CNC(=O)COC3CC3)CC2)=O)nnc(O)c2ccccc12 c1(OC)ccc(F)cc1CCC(=O)NC1(CCNC(=O)CNC(C)=O)CCC1 C(CS(=O)(=O)C1CC1)NC(CCN(C(C)=O)CC)=O c1(NC2C(C)CCN(C(=O)CCCCF)C2)cc(=O)n2cc(Cl)ccc2n1 c1(OCC(=O)NC2C(NC(c3cn(CSCC)nc3)=O)CCC2)ccccc1Cl O=C1OCc2c(NC(C3(F)CCN(C(=O)CN4CCNC(=O)C4)C3)=O)cccc21 c1(C(=O)NCc2cc(Cl)cc(Cl)c2)ccc(N=c2ccn3ncc(I)c3[nH]2)cn1 C=CCN=C(NCC(F)(F)C1CCC1)NCC(C)(F)F N1(C(C=C(C)C2CC2)=O)CCCC(C2CN(C(=O)C(F)=C3CCC3)C2)C1 S(=O)(=O)(CC(=O)NC1CCC(NC(=O)CSCC(N)=O)C1)NC C1(CNC(C(C2CC2)OC)=O)CN(C(=O)CCOCC2CCC2)CCCO1 c1(C(=O)OC)cnc2c(Br)cncc2c1NCC1CC2CCC1CN2 O=S(=O)(c1cc(Cl)cc(Cl)c1)N1CC2(CCN2Cc2ncccc2F)C1 C1(F)(CNC(c2cc(C)oc2C)=O)CCCN(Cc2ccncc2)C1 CCCCC(O)C(=O)NC(C)(C)CN(C)C(c1sccc1C(=O)OC)=O CC1=C(C(=O)N2C3C(NC(C4(C)CCCS4(=O)=O)=O)CC(C3)C2)SCCO1 c1(C(=O)NC2C(C(=O)NC(C(=O)OC)C(C)(C)C)C2)cccc([N+](=O)[O-])c1Cl Cc1ccc2c(c1)SC(C(=O)NCC(C1CC1)NC(c1cc(C(F)F)no1)=O)C2 C=CC1(C(=O)NC2CCC(CCC(N3CCC(COC)C3)=O)C2)CCCCC1 C1(CC(N2CCOCC(NC(C3(COC)CCC3)=O)C2)=O)CCC2(CCC2)CO1 C1(C(=O)NC2CN(C(CCC(=O)N(C)C)=O)CC2O)CC(c2ccccn2)=NO1 c1(OC)cccc(C(C)C(=O)N(C(C)CNC(c2cc(Br)c(C)s2)=O)C)c1 n1(CCC)nnnc1C(c1csc(Cl)n1)NCC(C1CCCCC1)OC n1(C(C(=O)NCCN(CC)CC)C)cc(CN2CCCC2CO)nn1 C1(CNC(=O)CC(F)F)CN(C(=O)Cc2csc(-c3ccc(F)cc3)n2)CCO1 c1(C(=O)NCc2ncn(C)c2)ccc(-c2ccc3ncsc3c2)c2c1OCO2 C1(NC(C(COC)N(C)C)=O)C2CC3C1C3C2c1nc(C2CC3(CCC3)C2)no1 Cc1cc(C(N2CCC(CCNC(C3C4CCCC34)=O)CC2)=O)c(Br)s1 c1(CC(C)(C)N(C(C23CC2C3)=O)C2CC2)cn(C(C)(C)C)nn1 c1(NC(C2N(C(CCOC)=O)C3C(C2)C3)=O)cc(F)c(Cl)cn1 CC1CN(Cc2sc(C(=O)NCC(F)(F)F)nc2C(F)(F)F)CC[SH]1C(C)(C)C Cc1c(C(=O)NC(CNC(C2CC(N(C)C)C2)=O)C(C)C(C)C)cccc1Cl CCC(C)CC(C)C(=O)NC(CNC(=O)Cc1ccc(F)nc1)C1CCC1 c1(CC)ccc(C(=O)N(CCC(C)NC(=O)C(c2ccc(Cl)nc2)(C)C)C)nc1 C1(C(=O)NCC2(OC)CC2)C2CCCC2CN1C(=O)CC1C=CCC1 C1(CNC(C2C(=C)C2)=O)CC2(CCC2)CN1C(=O)Cc1cnn(C(C)(C)C)c1 C#Cc1ccc(C(N2CC(NC(=O)CC(=O)N(C)C)C3(CC3)C2)=O)nc1 CCCC(O)CC(=O)N1CC(CNC(c2cc(CC3CCC3)c[nH]2)=O)C(O)C1 C(=O)(C1=NN(C)C(=O)CC1)NCCOCCN(C)C(C1CCCC1(F)F)=O C(=O)(CCC(C)(C)C#N)NC(C(=O)N(C)Cc1ncc(C)o1)Cc1ccco1 Cn1nc(C(=O)NC2(CCNC(=O)CC3CCNC(=O)C3)CC2)cc1CO C1(CN(C)C(C23C=CC(CC2)C3)=O)CCN(C(=O)Cn2cnnc2)CC1 C12(C(=O)NCc3ccc(NC(C(C)Oc4ccccc4)=O)o3)CCC(CC1)O2 CN1CCCC(O)(CC(=O)NCC2C3CN(C(c4cncn4C)=O)CC23)C1 N1(C(c2cn(C3COC3)nn2)=O)CCOC(CCN2CCSCC2)C1 CC(C)(CS(C)(=O)=O)C(=O)N1CCN(CCNC(=O)C(C2CCOCC2)F)CC1 N1(C(C2=NNC(=O)CC2)=O)CC(C2CCCCN(C(C3(O)CCOC3)=O)C2)C1 CCC(O)C(C)C(=O)N1CC(C)(NC(c2cccc(C(N)=O)n2)=O)C1 N1(C(CCNC(CC(C)C)=O)=O)CCC(C)(NC(=O)CCC2CCCCC2)CC1 Cc1ccnc(O)c1C(=O)N(C)CCN(C(=O)CC1(C)CCCC1)C N1(C(Cc2c(C)noc2Cl)=O)CC2(CCN(C(C3(CCF)CC3)=O)CC2)CC1C C=C1CC2(C1)CN(C(=O)C(CC)N(C(=O)C(C)(C(C)C)OC)C)C2 C(CC(O)CC(=O)NCCN(C(C1CCO1)=O)Cc1ccccc1)SC N1(C(C(C)CO)=O)CCCCC12CC(NC(=O)Cc1ccc3c(c1)CCN3C)C2 N(C(=NCc1cnc(C)cn1)N1CCCC(OCC2CCOC2)C1)CCC(CC)C N1(CC)CCC(NC(C2CC(=O)CN2C(C2CCCO2)=O)=O)CC1 c1(C(=O)NC2CCN(C(CC(C)C3CC3)=O)CC2)cccc([N+](=O)[O-])c1Cl Cc1cc(F)ccc1N1CCC(OC(F)F)C1.N12CCC(C1)NC2=O C1(CC)CCCC1(C)C(=O)NC1(C(=O)NCCC2CC(O)C2)CC1 c1(C(C(=O)NC2C(CNC(c3cc(C)ncc3)=O)C2)(F)F)cc(C)cc(C)c1 c1(C(N2CCN(C(C(c3ccccc3)C)=O)C(CF)C2)=O)c(Cl)ccc(F)c1N N1(CC)C(=O)CCC1CC(=O)NCC1C=CCN1C(=O)COc1ccccc1F N(C(=NCCC(C)SC)NCc1cc(Cl)ccc1C)Cc1c(C)cccc1 N1(C(CCC2CN(C(C3(C(C=O)CC)CCC3)=O)C2)=O)CCC(O)C(C)C1.OC C(=O)(C(F)(F)C(C)(C)O)NCC(CNC(CCC#C)=O)C(F)(F)F c1(NCCS(=O)(=O)CCO)ccccc1S(=O)(=O)NC1CC1c1ccccc1 NCCC(C(=O)NCc1csc(C2CCOCC2)n1)c1c[nH]nc1Br c1(NC(C2CCN(C(C3CC(=O)NCC3)=O)C2)=O)cccc(Br)c1[N+](=O)[O-] C#CCCCCC(=O)N1CCN(C(=O)C(C)OC(C)=O)CC1CCO c1(CNC(C2CCCC2C)=O)ccc(C(OC)OC)cc1.C(CC1CC1)CC CCCCC(CNC(C1C(Cl)(Cl)C12CC2)=O)NC(c1cnn(CC)c1)=O N1(C(CCN(CCCCC)C)=O)CCOCC12COCCN(C(=O)C=NOC)C2 c1(C(=O)NC2CCCC(NC(c3cn(C)nc3)=O)C2)cc(N)c(Cl)cn1 c1(C(=O)NC2CCN(C(c3[nH]c(=NCC)sc3)=O)C(C)C2)cc(C)c(Cl)cc1C N1(C(C(COC)Cl)=O)CC2CCC(C1)N2C(=O)CN1CCCNC1=O N1(C(CC2CC(CC)C2)=O)CC(NC(=O)CNC(=O)OC(C)(C)C)C(SC)C1 c1(C(=O)NC(CC)CNC(C2(CO)CCOCC2)=O)cc(OC)cc(N)c1O N1(C(C(CC)COC)=O)CCCC2C1CCN2C(c1cc(C)cc(C)n1)=O N1(C(COc2ccc(C)cc2)=O)CCCC2C(NC(c3ccns3)=O)C(C)(C)C12 C(=O)(CC(CC)CC(C)C)NC(CC=C)CNC(c1cc(C(C)(F)F)on1)=O CC(C)CCC(O)C(=O)NCC1CC(NC(c2c(O)cc(Cl)cc2Cl)=O)C1 c1(C(N2CCC(N(C(=O)C(CC)CC=C)CC#C)CC2)=O)cc(C)c(C)cc1Cl Cc1[nH]nc2c1CN(N1CCCCC1C1CCCC1O)CC2 c1(C(C(=O)NCC(C)N(C(C2COCCO2)=O)CC)C)ccc(C(N)=O)cc1 Cc1ccc(C(=O)NC2CC(C)N(C(C3C(C)C3C)=O)C2)c2c1CCC2 C1(NC(C(CC)=CCCC)=O)CC2(CCC(NC(=O)CCS(=O)(=O)NC)CC2)C1 C1(OC)CCN(C(=NCCc2ccc(OC)nc2)NCc2cc(C)on2)CC1C CCC(CC(=O)N1C2CCC(C2)C1CNC(c1ccncc1C(F)F)=O)C(C)C Cc1cccc(C(=O)NC(C(C)NC(C2(C)CCC2)=O)C(C)C)c1 N1(C(C=CCOC)=O)CC2CCC(C1)N2C(c1cc(C(C)(C)C)n[nH]1)=O C(C(C(=O)NCC)Nc1ccc(CC)o1)SCC=C Cc1nn(C)c(C)c1C(=O)N(C1(C(N2CCC(C#N)C2)=O)CC1)C CC1(C)CC(CC(N2CC(O)(CNC(C3(C)CCNC3=O)=O)C2)=O)CC(C)(C)O1 N1(C(c2cc(F)c(I)c(F)c2)=O)CCC2(CCN(C(C3(F)CC3)=O)C2)C1 C1(C(N(C(C)C(C(=O)CCc2cc(N)no2)=O)CC)=O)CCC(C)C1.OC C1(NC(C2C(C)(C)C2)=O)CN(C(=O)CCSC(F)(F)F)C(C)(C)C1 c1(CC(=O)N(CCN(C(C(C)N(C(C)=O)C)=O)C)C)ccc(C(=O)OC)nc1 c1(-c2ccc(C(=O)NC(CN(C(=O)COCCCF)CC)C)s2)cccc(F)c1 c1(C(N(CC(=O)NC2CC2)CC#C)=O)ccc(C)cc1CC.C(CCN(C)C)N.C N1(C(c2c(C)occ2)=O)CCCC(NC(=O)CCc2ccc(Cl)cc2Cl)C(F)C1 CCCC(C(=O)N1CCOC(CCNC(N2CCOC2=O)=O)C1)NC(C)=O.CC C1(C(C)NC(=O)CCCN(C)C)CCCN(C(=O)C(CCN(C)C)N(C)C)C1 Cn1nnc2cc(C(N3CC(CNC(C4CCOCC45CCC5)=O)C3)=O)ccc12 c1(NC(C2CCCN(C(C(C)C(F)(F)F)=O)C2)=O)cnc2c(c1)CCC2 N1(C(c2cc(SC)c(Br)cc2)C(=O)NCC2CCOC2)Cc2cc(O)nnc2C1 C1(OCC(=O)NC)CCC(N2CCCC2=O)CC1.c12nc(no1)C2 CC1(C)CC(CNC(=O)CCc2cnco2)N(C(C2CCC2(C)C)=O)C1 C1(C(=O)OC)CCC(C(N2CC(CNC(=O)CNC(N)=O)C2)=O)C1 N1(C(CC(C)C)=O)CC(O)CC1C(=O)NCC12CC(C(N)=O)(CO1)C2 C(=O)(C(C(C)OC)NC(C1CC1(Cl)Cl)=O)OCC Cn1cc2ccc(C(=O)NCCC3COCCN3C(=O)Cc3ccsc3)cc2n1 N1(C(C(C=CC)O)=O)CC2(CCN(C(c3cccc(O)n3)=O)C2)C1 Cc1cc(Br)c2c(c1)CN(C(=O)NC(c1ccc(OC(F)F)cc1)C)CCO2 C1(ONC(c2occ(C(=O)OCC)c2)=O)CCC(=O)NC1=O C(=O)(CC(C)(C)N(C(=O)C(C)CC#N)C)NCC(C)OCC=C C1(N(c2cccc(-n3ccnn3)c2)CC#CN(C)C)CCCC(=O)CC1 CC(C)CC(C(=O)NCCc1ccncn1)NC(=O)C(C)O c1(OCC)ccc(CC(N2CCC(N(C)C(c3nc(=O)n(C)[nH]3)=O)C2)=O)cc1 c1(C(=O)OC)cc(C)nn1CC(=O)NC1CCC(CNC(=O)C=CC2CC2)C1 N1(C(C(CC)C(C)O)=O)CCC(C2(NC(=O)C=Cc3ncccc3C)CC2)C1 c1(OC)cc(N)ccc1NC(=O)C(=O)NCC1(C(F)(F)F)CCCCCC1 C1(CC(=O)N(C(c2cn(CC3CC(F)CN3C)nn2)C)C)SC2=NCCN2C1=O C(C(=O)NOCC(=O)OC(C)C)(c1ccccc1)NC(C=CC(CC)C)=O C1(NC(c2c[nH]cc(C)c2=O)=O)C2CC3CN(C(C4CCCS4)=O)C1C3C2 C1(C(N(CCCNC(c2c(CCC)occ2)=O)C)=O)CC(=O)N(C(C)CCC)C1 N1(C(CCCC(N)=O)=O)CCCC2(CNC(=O)C(F)C3CCCC3)CCCC12 C12(CNC(c3ccn(CC)n3)=O)CCC(C1)N(C(=O)CCC(C)(C)O)C2 C1(C)(CNC(c2n(CC)ccn2)=O)CN(C(=O)C(C)c2ccsc2)C(C)(C)C1 n1(CC(=O)NCCOCCC(=O)N2CCCC2)cccnc1=O.C12CCC1C2 C1(CNC(C(=O)NCCNC(C)=O)=O)CN(C)CCN1C(=O)C(C#N)C(C)C Cc1cccc(CNC2(C(=O)NCC(C)O)CC2)c1 c1(N2CC(C)=C(C)CC2)nc(=N)[nH]c(=NC(C)Cc2ccc(Cl)cc2Cl)[nH]1 c1(CC)n[nH]cc1C(=O)NCC1CC(C(=O)NCC2CC(CN=[N+]=[N-])C2)CO1 c1(-c2scc(OC)c2)ccc2nccc(C(=O)Nc3c(F)cc(F)cc3Cl)c2c1 C1(NC(CCC(=C)C)=O)CS(=O)(=O)C12CCN(C(C1(C)CCCS1(=O)=O)=O)CC2 C=C=CC(C)C(=O)NC(C)(C)CCN(C(=O)Cc1cc[nH]n1)C Cc1nc(C(C)(C)C)nc(O)c1C(=O)NC(C)C(CO)NC(=O)C#CC1(C)CC1 C1(C(=O)NCC(=O)N(CC)CC)Cc2nccn2C1.C(C)(C(=O)O)N N1(C(Cc2c(C)noc2)=O)CCC(NC(c2ccc(C(C)C)c(Cl)c2)=O)CC1C C1(C(=O)NC(CNC(C=C(CC)CC)=O)C)CC(C)(C)C12CCC2 O=S(=O)(c1cccc(=NCCN2CCCC2)[nH]1)NCC1CCC2CC12 C(c1ccc(C)cn1)=CC(N1CC(CCO)(NC(C(CC)n2ccnc2)=O)C1)=O N1(C(C(CCC)C(C)C)=O)CCC2C(CCN2C(c2cccc[n+]2[O-])=O)C1 C=C=CCC(=O)OCCOCCCCOCC(C)(C)C C(C(C)(C)C(=O)N1CC(CC(F)C(=O)NC2CCC(CN(C)C)C2)C1)SC CCCCCCC(C)CC(=O)N1CCC(NC(c2cnn(C(F)F)c2)=O)C(O)C1 C1(NC(c2c(C)oc(Cl)n2)=O)CS(=O)(=O)N(C)C12CCN(C(=O)CO)CC2 Cc1cccc(C(F)(F)C(=O)NCC(C)NC(=O)Cn2nnc(=O)[nH]2)c1 C(CC(=O)N=c1ccn(C)[nH]1)N(CC#C)C(C1CCC(C)(C)OC1)=O C(=O)(C1CCCc2nccn21)N(S(C)(=O)=O)C.C12(CCC1)CN2.C12(CC1)CC(=O)N2 c1(OC)cc(NC2CC(NC(C3(C)CC3Br)=O)C2)ccc1[N+](=O)[O-] C1(C)(CC)CCN(C(c2ccccc2N(C)C)C(=O)NC2CCOC2)C1 C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCCCN(C(c1ccc(C)nn1)=O)C Cc1nc(C2CC2)ncc1C(=O)NC1CC2(C1)CC(NC(C1CCC1CF)=O)C2 c1(N(C(C(C)O)=O)C)cccc(CNC(C2(CCC(F)(F)F)CC2)=O)c1 c1(C(N(CCN(C(c2c(C)cc(CC)o2)=O)C)C)=O)nccc2ccccc12 c1(C(=O)NCCC2(NC(CC(C)n3ccnc3)=O)CC2)cccc2c1CCC2 c1(C(N2C(CN(C(C(CC)N(CC)CC)=O)C)CCC2)=O)cc2c(ccn2C)[nH]1 CC1CCCN1CC(=O)NC(c1nocc1C(=O)NC1(CCCCO)CC1)C N1(C(C23CC(n4cc(C5CCN(C)C5=O)nn4)C2C3)=O)CC2(CCOC2)C1 Cc1nnc(NCC2CCC(CNC(c3ncccn3)=O)CC2)c(C#N)c1C c1(C(C(=O)N2CC(NC(=O)COCCF)C2)SC)ccccc1C(F)(F)F C1(NC(CC2C(NC(c3cnc(C(C)C)o3)=O)CCCC2)=O)CCC(C2CC2)C1 CCC1=NOC(CC(=O)NCC=CCC(=O)N(CCOC)CC)C1 C(=O)(CC1OCc2ccccc21)NC1C(C)CN(c2ncccc2C#N)CC1 CC1C(C(=O)N2CCC(CO)(CO)C2)=C(C)NC2=C1CC2 C(c1ccc(F)cc1)=C(C)CN(CCC(O)C(C)(C)C)C Cc1coc(C2CCCN2CCCn2cc(CNC(N(CCCO)C)=O)nn2)n1 C1(NC(Cc2ncn(C)c2)=O)CN(C(=O)CCN2CCC(F)C2)CC1N=[N+]=[N-] N1(C(C2CC(C#N)C2)=O)CC2CC(NC(c3cc(F)cc(F)c3)=O)C1C2 c1(OC)ccc(-n2cc(CNC(=O)Cn3nnc(C4CC4)n3)nn2)cc1 C(CC(=O)NC1CC(NC(C2CC2OC(C)(C)C)=O)C1)NC(C)=O CC1CC(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)CCS1(=O)=O N1(C(C(C)(C)c2ccns2)=O)C2CCC1CN(C(=O)COC1CCC1)C2 c1(OC)ccc2cc(O)c(-c3sccc3C(N3CCCCNC(=O)CC3)=O)cc2c1 CC(C)C(C(=O)NC(CNC(c1cnc(C2CCC2)s1)=O)C1CC1)n1cnnc1 C1(CCN(C(C(C)OC)=O)C)CCN(C(c2ccc(C(F)(F)F)cn2)=O)CC1 Cc1cc(C(N2CCC3(NC(c4cnc(C(F)F)nc4)=O)CC3C2)=O)c(C)n1C Cc1cnn(CCN(C)C(C2CCC2NC(C2CCN(C3COC3)C2)=O)=O)c1 C(C(C(=O)NCCC1CCN(C(=O)C=CCn2cncn2)C1)OC)OC C1(NC(c2n(C)c(O)nc2)=O)CC2CN(C(C3CC=CC3)=O)CC2C1 C#Cc1ccc(F)c(C(=O)NCC(CNC(c2c[nH]nc2C(C)(C)C)=O)CO)c1 N1(C(c2cc(C)sc2C)=O)CCC(NC(=O)C2=CSCS2)C(F)C1 C(=O)(C(=O)CC(C)CC)NC1C(C(N2CCCC(CC)CC2)=O)OCC1 C12(C(=O)NC(c3ncc[nH]3)CC)CC(CN1C(=O)CC(C)OC)C2 C1(NC(C2C(C(C)(F)F)C2)=O)CCCN1CC(=O)NC(C1CCCC1)C1CC1 CC1C2CCC(C2)C1C(N1CCC(OCC(=O)NC2CN(C3(C)CC3)C2)CC1)=O C1(CCC)CCC(C(=O)NC(=O)C(C)Cc2ccccc2)CC1 C1(C(CNC2(c3onc(C(C)C)n3)CCC2)C)OCCCC1(C)C c1(C(N2CCC(CC=C)(NC(=O)C(C)C3CCCO3)C2)=O)c(C)ncnc1C C(C)(C(=O)N1CCC(C)(CNC(=O)Cn2cc(Cl)cn2)C1)(C(C)C)NC(C(C)C)=O CC(C)CC(C)CC(=O)NCC1COCCN(C(=O)C#CC(=O)N(C)C)C1 C(=O)(C1=CCOCC1)N(C)CC1CCN(C(c2nn(CC)c(C3CC3)c2)=O)C1 N1(C(c2c(C)ccc(C)n2)=O)CC2(CC(C(=O)NC(CO)CC(C)(C)C)CO2)C1 C1(OC(C)C(=O)NC2CCC2NC(c2ccc(=N)[nH]n2)=O)CCCCCC1 Cc1cccc(C(N2CCCC2Cc2cn(CC3CC4CCC3O4)nn2)C)c1 c1(C(CO)NC(C2CCN(Cc3cnccc3Cl)C2)=O)ccc(Cl)cc1 N1(C(c2cccc(CC)c2O)=O)CCC2(CC1)CC2NC(=O)CCC(F)(F)F c1(CN2CCN(C(=O)C(Cl)(Cl)Cl)C(CO)C2)c[nH]c2c([N+](=O)[O-])cccc12 CC(C(=O)N(C)CC1(NC(=O)C=CCC2CC=CC2)CC1)N1CCCC1 N1(C(C2(C)COC2)=O)CCC2CCCN(C(=O)CS(C)(=O)=O)C2C1 C(c1ccccc1C)=CC(=O)N(C1CCN(C(C(C2CCC2)OCC)=O)C1)CC c1(CC(C)NC(C(C2CCC2)OC)=O)ccc(C)cc1Br c1(NC)ccc(C(N2CC3C(NC(C4(NC(N)=O)CC4)=O)C3C2)=O)nc1 c1(C2C(C(=O)NCCCN(C)C(C3CCCSC3)=O)C2)cccc(Br)c1 N1(C(c2cc(C)[nH]n2)=O)CC2(CCCC2NC(c2occ3c2CCOC3)=O)C1 C(N=c1cc(NCCCCN2CCCC2)nc[nH]1)C1(N(C)C)CCSC1 CCCCCCCCNC(C1CC2(CCN1C(=O)CCCN1CCCC1)CC2)=O C(=O)(CCC(C)C)NCCNC(C(C)(C)N(C(COCC)=O)CC)=O.C(C)=O CC1(C)CCC(CN=c2nnc(C(F)F)c[nH]2)(NC(C2CCCC(=O)N2)=O)CC1 N1(C(CCS(=O)(=O)N(C)C)=O)CCC2(CC(NC(C3C=CCCC3)=O)C2)C1 N1(C(C(C)(C)c2cncs2)=O)CC2CCCC(C1)N2C(=O)CN1CSCC1=O C(=O)(CC(O)CCCCC)NC1(CC=C)CCN(C(c2cnn(C)c2C)=O)C1 C1(NC(=O)OC)CCN(C(=O)CSC2C3CNCC23)CC1 Cc1cc(Cl)c(C(=O)NC2CCN(Cc3ccc(C)c(C)c3)CC2O)cn1 c1(C(N2CCN(C(c3cn(C(C)C)nn3)=O)C(C)C2)=O)cc2cccc(Cl)c2s1 C1(C#N)(C(N2CCC(O)(CNc3ncc(C)cn3)CC2)=O)C(C#N)C1(C)C C12(NCC3(CC)CCOC3)CCC(C(=O)NC3(C)CCC3)(CC1)CC2 c1(C(=O)NCCN(CCC)C(C2(COC)CCCC2)=O)nc(Cl)c(CCOC)[nH]1 C1(F)(C(N2CC(OC)C(NC(=O)C(C)C3CC3)C2)=O)CCN(C)CC1 c1(-c2cn(CC(=O)NCCc3cc(C)no3)nn2)ccc(SC2CCCC2)cc1 N(C1Cc2ccccc21)C(CC1CCN(c2cncc(C#C)n2)C1)=O C1(C(=O)NC(C(C)C)CCNC(C2CC(=O)NC(=O)N2)=O)CCc2cnnn2C1 N(C1CCCc2c1cnn2C)C(C(=O)N(C1CCCC12CC2)C)=O C(=O)(CC(C)(C)C1CCCCC1)N(C1CC(NC(=O)C=Cc2ccncc2)C1)C c1(C(N2CCC3CN(C(C4C(CN(C)C)C4)=O)C3C2)=O)cc([N+](=O)[O-])cnc1O C(C(=O)NCCCn1cncn1)(C(C)C)SCC.C1(C2CCC2)C(=O)N1 N1(C(C2(C(=O)NC)CC2)=O)CCC2(CC1)CC2C(=O)NCCC1CCCCCC1 c1(N(C(C2CCCC2(C)C)C(=O)NCC(=C)C)C)ccc(OC)cc1C C1(C2CCN(C(=O)CCP(C)(C)=O)C2)(NC(C(C)OCC)=O)CC1 N1(C(C(C)(C)CN2CCOCC2)=O)CCC(O)(CNC(=O)COC(=O)C2CC2)CC1 CCCC(C)(C)C(=O)N1C(CNC(=O)Cn2c(C)c(C)sc2=O)CC2CC12 N1(C(CCc2ccn(C)c2)=O)CCCC(C)(C)C1CNC(C1(C)CCNC1=O)=O Cc1nc(C)c(C(=O)NC2CCC(NC(C3CC34CCCC4)=O)CC2)s1 c1(C(=O)NC2CCC(N(C(c3c(C)cccn3)=O)C)C2)cc(N)cc(O)c1C C1(CCNC(COCCOCC#C)=O)CCCN(C(=O)CC2CC3CC3C2)C1 N1(C(c2scc(C)c2)=O)CC2(CCNC(c3ccc(Cl)cc3)=O)CCC1C2 Cc1noc2ncnc(NC3CC4CN(C(=O)CSc5cccc[n+]5[O-])CC34)c12 C(CC(C(=O)NCc1ccc(Cl)cn1)NC(=O)CCOC(C)C)=CC CCCCC(CN=c1[nH]c(C)nc(C)c1F)NC(c1ccncn1)=O Cc1ccc(C(N2CC(C(N3CC4C=CC3CC4)=O)C(F)(F)C2)=O)cc1C#N N1(C(C(Cn2ccc(C)n2)C)=O)C2CCC1C(C)C(NC(=O)CC1CN(C)C1)C2 Cc1cc(Br)sc1C(=O)NCC(C)NC(=O)CCc1ccco1 CCCC(CCC)C(=O)NCc1nc(C(N2CC(COC)C2(C)C)=O)co1 N1(C(c2c(C)cccn2)=O)C2CC=C(C(=O)N3CC(O)(c4nn[nH]n4)C3)C1CC2 c1(OC)cc(CO)ccc1C(=O)NC1CCC1CNC(c1nn(C)c(C)c1Cl)=O NS(=O)(=O)c1coc(C(=O)NC23CC(C2)N(C(c2cn4ccccc4n2)=O)C3)c1 c1(C(CC(=O)N(CC(C)NC(=O)C(F)=CCCF)CC)C)cccc(F)c1 c1(C(N(CC(=O)NC2CC(CCF)C2)CC2CC2)=O)cocc1C(N)=O c1(NC(C2C(NC(c3ccccc3COC)=O)COC2)=O)c(C(N)=O)c(C)nn1C c1(OC)cccc(Cl)c1C(N1CCC(NC(c2nc(C)ncc2Br)=O)C1)=O C12(OC)CCCC(CC(NC(=O)Nc3ccc(SC)nc3)C1)C2 N1(C(COCC#C)=O)CCC(N(C)C(c2c(Br)noc2C2CC2)=O)CC1 N1(C(c2c(OC)cnnc2)=O)CC(C)CN(C(c2cncnc2C)=O)CC1C C=CCCC(C)N=c1nc(N(C)CC2CCOCC2)c2c([nH]1)c(C)nn2C C1(CNC(CCN(CCC)C)=O)CC2CCC(C1)N2C(=O)C(C(C)OC)N(C)C C1(C(=O)Nc2cn(COC)nc2)C2CC1N(C(c1ccc(Cl)cn1)=O)C2 c1(C(=O)NCCCOCCCNC)cc(S(C)(=O)=O)c(C)o1 c1(CC#N)ccc(C(N2CC(NC(c3cc(C4CC4)ccn3)=O)C(O)C2)=O)cc1 c1(NC(C2(C(=O)Nc3nc4ccccc4o3)CC2)=O)ccc2c(c1)CCNC2 N1(C(c2cn(CC=C)nc2)=O)CCN(C(c2csc(Cl)n2)=O)CC(O)C1 C=C1CCC(C(N2CC=CC(NC(=O)C(C)CSc3ccccc3)C2)=O)CC1 C1(NC(C(COC)COC)=O)CCCCN(C(=O)C=Cc2ccccc2)C1 c1(C(=O)NC2C=CCN(C(C3CCC(C)(C)CC3)=O)C2)ccc2cnoc2c1 C1(C2N(C(c3ncc(CC)s3)=O)CCC2)CCN(C(=O)CN2CCN(C)CC2)CC1 C1(NC(C2N(C(C34CCC(OC)C3C4)=O)CC2)=O)Cc2cccnc2C1 Cc1cc[nH]c1C(=O)NCCCCCNC(=O)C(C)NC(=O)Cc1ccccc1 N1(C(C2(NC(CCn3c(C)nnn3)=O)CCC2)=O)CCC(C(C)CO)CC1 CCC(CC(=O)N1CCCC(NC(=O)Cc2ccn(CC)n2)CC1)C(C)C C1(C(=O)NC2CC(NC(C(C)NC(=O)C3CC3)=O)CC2O)CCCC12CCC2 c1(C(=O)NCC(C)N(C)C(c2sccc2OCC(F)(F)F)=O)cc(O)ccc1F Cc1nc(C(C)C)sc1C(N1CCC(CNC(c2c[nH]nc2Cl)=O)C1)=O n1(CC)nc(C)c(CC(N2CCOCC(NC(=O)CC(C)O)C2)=O)c1C N1(c2ncc(C#C)cn2)CC2(CN(C(c3cccnn3)=O)CC(C)(C)O2)C1 CC(CF)C(=O)NCCC1CCCN1C(c1ncn(C(C)(C)C)n1)=O c1(CN2C(CN3CC(C)OCC3)CCC2)ccc(O)c(C(=O)O)c1 C1(N(c2ncnc(N3Cc4cccc(C)c4C3)c2C)C)CCCCC(S(C)(=O)=O)C1 C=CCC(C)(CC)C(=O)NCc1ccc(C(=O)NCc2ncccc2C)s1 C(=O)(C(CCC)OCC)NCC(CNC(C1(C=C)CC1)=O)CO CCCCC(CC(=O)NCCCC1CC=CCC1)NC(c1cccc2ccoc12)=O N1(CC)CC(C(=O)NCCC2(CNC(c3cnn(CC(F)F)n3)=O)CC2)CC1=O N1(CCC(=O)NCc2cn(CC(=O)NCC3(CO)CC3)nn2)C(=O)CCC1=O CCC(C)C(C(=O)N1CCCC(CCNC(=O)CCCCSC)C1)OC N1(OC)C(=O)C2CCCCN2C1=O.C1(CC(=O)OC)CC2N(C1)C2=O Cc1onc(-c2ccc(F)cc2)c1C(=O)NCCn1cc(C2CCCN(C)C2)nn1 c1(C(=O)NCC(C)NC(C2(F)CC3CC2C3)=O)cncc2sccc12 C1(NC(c2cnc(SC)s2)=O)CCC(C)(CNC(=O)CCc2cccn2C)C1 N1(C(CC2N(C)CCCC2)=O)CCCOC(CNC(=O)Cn2cnnn2)C1 Cc1ccc(C(=O)NCCCC2(NC(C3(C)CCC(=O)N3)=O)CC2)c(F)c1C c1(NC(C2(F)CCN(C(Cc3nc(C)on3)=O)C2)=O)cc(C)cc(Br)c1F N1(C(c2c(CC)ocn2)=O)CCN(C(=O)C(C(C)(C)C)NC(N)=O)C(C)C1 C(CN=c1c([N+](=O)[O-])c[nH]c2c(Cl)cccc12)=CCNC(=O)CCN1CCC1 C1(C(=O)NCCC(C)NC(=O)CCc2ccc(F)nc2)C2C3CCC(C3)C12 C1(N2CC(CC3(C)CN(C(C45CC(C(=O)O)(CO4)C5)=O)C3)C2)CCCN1C=O C1(NC(Cn2c(C(C)C)ncc2)=O)CN(C(=O)C2=CC(C)(C)C2)CC(F)(F)C1 c1(NC(C(C)NC(C)=O)=O)cccc(NC(=O)C(C)(C)CN(C)C)c1 C(CC(F)F)(C(=O)NC1CC(C)(C)C12CC2)NC(Cc1c(C)n[nH]c1C)=O Cc1ccc(C(=O)NCCC2CCC(NC(=O)C(=O)NCC(F)(F)F)C2)s1 c1(OCC)cc(C(N2CCC(N(CCO)C(C34CC(O)C3C4)=O)C2)=O)[nH]n1 N1(C(C(C)Oc2ccccc2)=O)CCN(C(C2CC3(CC(=O)N3)C2)=O)C(C)C1 CC1(C)CCCCC(C(N2CCN(C(C3C4COCC34)=O)C(CCO)C2)=O)C1 CCC(C)C(C(=O)N1CC2CC1CN2C(c1csc(F)c1)=O)N(C)C C1(NC(C(C)O)=O)CC1C1CCCN(C(c2cn(C)nc2C2CCC2)=O)C1 N1(CC=CC(=O)N(CC(CC)NC(=O)Cc2csc(S)n2)C)CCOCC1 c1(C(=O)NCC2(CNC(C34CC(C)(C3)C4)=O)CCCC2)cc2n(n1)CCNC2=O c1(CNC(C2(CCC)CCC2)=O)cc(C(=O)NC2CC(N3CCCC3)C2)n[nH]1 c1(C(N(CCCCN(C(c2cnc(C)s2)=O)C)C)=O)cccc(-n2cncn2)c1 N1(C(CCOC(C)C)=O)C2CCCC1CN(C(C1CC=CCC1)=O)CC2 CC1(CC(=O)NCC(O)CCNC(=O)CCSc2ccccn2)OCCO1 C(CC(O)C(=O)N1CC2CC2(C(=O)NCc2nnc(C)o2)C1)SC CC(C)(F)C(C)(F)C(=O)NCC1CC(C(=O)NOC2CCC2)C1 Cc1cc(C(=O)N(CCCCN(C(=O)C(C)CO)C)C)oc1C c1(NC(CCC)C)ccc(S(=O)(=O)N2CCCC2c2ccc(OC)cc2)cc1F C1(CN(C(=O)C2=CCC2)CC2CC2)CCN(CC(=O)NC2(COC)CC2)C1 CC(O)C(C(N)=O)NC(=O)CCC1CCCN1C(C1CC12CC2)=O N1(C(CC(n2ccc(C)n2)C)=O)CCCC2(CCN(C(=O)C(C)CN(C)C)C2)C1 N1(C(COCCCCC)=O)CCC(C(C)C(=O)N2CCC2c2cnn(C)c2)CC1 CCC(CC)C(C)C(=O)N1CC2CCCC2(NC(c2cnc(Cl)[nH]2)=O)C1 c1(N2CCCN(C(CCNC(COC)=O)=O)CC2)ncccc1S(C)(=O)=O c1(CC)cccnc1C(N1CC(O)CC1CNC(=O)C=CCF)=O c1(C(=O)NC(C2CN(C(=O)CC3CCNC3=O)CCO2)C)ccnc(CO)c1 C1(COC)(NC(c2sccc2SC)=O)CCN(C(=O)CC2C(=O)NN=C2C)C1 C(=O)(CC(O)C(C)C)NCCC1CC(NC(Cn2ccc(C)n2)=O)C1 C1(CNC(CCc2n(C)cnc2)=O)CCC2(CN(C(=O)C=CCO)C2)O1 c1(C(=O)NC(C2CCN(C(C3N=C(C)SC3)=O)CC2)C)c(Cl)ccc2ccoc12 c1(C(=O)NCC2COCCN2C(C2CCC(=O)N2)=O)cccc2c1CCC2 C(=O)(CS(=O)CCC(F)(F)F)N(C)CCN(C)C(c1cnc2nccn2c1)=O c1(CC(C(=O)N(CC#C)CC=C)NC(C2CNC(=O)O2)=O)ccc(Cl)cc1Cl N1(C(C2CCN(CC)C2)=O)CC2CCC(CNC(C3(SC)CC(=O)C3)=O)C2C1 C(=O)(C(CCC)CC(C)C)NCC1(OC)CN(C(c2cn(CCCC)nn2)=O)C1 c12ccccc1CN(CC)CCO2.C(=O)(C(O)CC1CCCCC1)NCC C1(C(N(C2CC(OC)C2)C)=O)CN(C(=O)CN=[N+]=[N-])C(C)(C)C1 N1(C(c2ccc[n+]([O-])c2)=O)CCC2(CCNC2)CC1 c1(NC(=O)NCC2CCC3CC23)cc2c(nc1O)CCCC2 N1(C(C2(C(=O)OCC)CC2)=O)C2CCC1CN(C(C13CCOC1CCOC3)=O)CC2 CC(C)C(C)C(=O)N(C)CC1CCCCN1C(=O)CC(=O)NC1CC1 C(=O)(C1CCc2cc(F)ccc21)NCC(CO)NC(c1c(C)n2c(n1)scc2)=O Cc1noc(CNC(=O)NCc2nc(C(C)O)n[nH]2)n1 C(c1ccccc1OC)=C(C(N1CCC(N(C(C2CC2(C)C)=O)CC)C1)=O)C C(C(=C)CCNC(=O)C(C1(O)CCC1)SC)NC(COCCCC#C)=O.C(C)(=O)O c1(N(C2CCNCC2F)C(c2ccc(C)cc2Cl)=O)ccn2nccc2n1 c1(C(N2C3(CN(C(CC45CC(C)(OC4)C5)=O)C3)CC2)=O)cc2scc(Cl)c2[nH]1 CC1CCN(C(=O)CNC=O)CC1NC(=O)CNC(=O)CCCCO Cn1nccc1C1CC1C(N1CCC(CN(C(C2CC(CF)C2)=O)C2CC2)C1)=O N1(C(C2CCN(CCC(=O)OC)CC2)C(=O)NCCC)CCCCC1CO N1(C(C2N(CC)CC2)=O)CCCCC1CN(C)C(c1ccc(OCF)cc1)=O C1(NC(C#CCNC(c2cccc(OC)n2)=O)=O)CCN(C)C(=O)C1 C=CC1CC(N=c2ccc(Br)c(S(=O)(=O)N(CC)CC3CC3)[nH]2)C1 C1(NC(CC(c2cccc(F)c2)C)=O)CCC(NC(=O)COCC(=O)O)CC1 CN1CCCC(O)(CC(=O)NCCNC(C2(CF)CC2)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NCC(CC(C)C)NC(CS)=O.Cc1cccc(C)c1 CN1C(=O)CCC1C(=O)NC(C(=O)NCCCOCCO)C1CC1 c1(NC(C2(O)CCN(Cc3c(Br)ccnc3Cl)CC2)=O)cc(F)ccc1[N+](=O)[O-] CCC(CC(=O)N1CCC1CC(=O)N(C(CO)CCSC)CC)C1CCC1 CC1(C(N2CC(NC(c3cccn4nnnc34)=O)C2)=O)COc2ccccc2O1 N1(C(c2cnn(CC)n2)C(=O)NCCC)C2CCCC1CC(F)(F)C2 S(=O)(=O)(c1ccc(NCC(C)(C)C)c(C#N)c1)N(CCn1ccc(C)n1)C C1(NC(c2cccc(CNC(C(C(C)C)(C)O)=O)n2)=O)CC2CCC(C1)C2O c1(C(N2CCCC(CC=C)(NC(=O)C3=NOC(C)C3)C2)=O)cccc(S(C)=O)c1 C(CC(=O)CCCC(=O)O)N(C)CCF.S(=O)(=O)(c1cccs1)N S(=O)(=O)(c1cccc(C(=O)NC(CNC(C2CC(C(F)F)C2)=O)C2CC2)c1)NC Cn1cc(S(=O)(=O)NCC(=O)NCCNC(c2cc3[nH]ccc3s2)=O)cn1 N1(C(c2c(OC(C)C)nccc2)=O)CC2CN(C(=O)COC3CCCCC3)C2C1 C1(OC)(CNC(C2(c3cccnc3)CC2)=O)CCCN(C(=O)CC(C)C(F)F)C1 C1(C(=O)NCC)(CNC(N2C(C(=O)OC(C)(C)C)C(CC)C2)=O)CC(F)(F)C1 c1(C(=O)NC(C)CNC(=O)CN(C)Cc2ccccc2)ncccc1S(C)(=O)=O C(=O)(CC(C)CC(C)C)NC1CC2(CC(NC(C=Cc3c(C)ncs3)=O)C2)C1 CCCCC(F)C(=O)N1CCCC(NC(=O)CCN(CC)CC)C2CC12 C1(NC(c2ccc(OC(F)F)cn2)=O)CC2CN(C(C3CCCCCC3)=O)CC12 c12ccc(Br)c(c1)NC(=O)C2N1CCC(c2ccc(Cl)nc2)C1.C(=O)(NC)OC N1(C(=O)NCCCOC(C)C)CCN(Cc2ccccc2)C(C)C1 C12(NC(CONC(=O)Cc3ccc(O)cc3)=O)CCC(CC1)OC2 C1(C(N2CCOCC2)=O)CC(O)CN1Cc1ccnc(-c2cccc(F)n2)c1 c1(C(C)O)cn(C2CN(C(C3(C)CC3C(=O)N(C)C)C)C2)nn1 C1(NC(c2[nH]cc(C)c2)=O)CCC(C(=O)N(C2CCCC2C)C)CC1 C1(NC(c2cnn(CC)c2Br)=O)CCCC12CCN(C(=O)CNC=O)CC2 c1(C(N2CCCCC(NC(C3CC(=O)N(O)C3)=O)C2)=O)cc2cnccc2[nH]1 c1(OC)cc(F)ccc1CC(N1CC(O)CC1C(=O)NCC1CN(C)CCO1)=O c1(SC)cc(C(N2CCCC2CN(C)C(C2CCO2)=O)=O)c(Cl)cc1Cl CC(CNC(=O)C(C1CCC1)NC(c1ccns1)=O)CCCO Cn1c(CNC2CCCC2C(=O)Nc2cncc(Br)n2)nnc1S c1(N(C)C)ccc(F)c(C(=O)NC2CC3CC2CN3C(=O)C2=CCCC2)c1 N1(C(C(C)SC)=O)CCN(n2cc(C(=O)N(C)Cc3c(C)noc3C)cn2)CC1 C1(C)(C(N2C(CNC(C=CCCC)=O)CCC2)=O)CC2CCC1CC21OCCO1 c1(OC)ccc(-c2ccc(CN(C)C)s2)cc1F N1(C(C(=Cc2cccs2)C)=O)CCC(C)C(NC(c2cnc(C)[nH]2)=O)C1 C1(CNC(C(C)=C2CCC2)=O)C(C)CCN1Cc1cccc(C)n1 C12(C(=O)NCC3(C)CCCN(C(C=CC)=O)C3)C3C4C1C1C2C3C41C(N)=O C1(N(C(C2C=CCCC2)=O)CC)CCN(C(c2sccc2OC)=O)CC1 Cc1cc2nccnc2cc1C(=O)NC1CCCC1NC(C1CC(C)(F)C1)=O C1(O)(CNC(c2cnc(C3CCOC3)s2)=O)CN(C(c2cn(CCF)nn2)=O)C1 Cc1c(F)ccc(Br)c1C(N1CC(N(C(=O)C=Cc2cncnc2O)C)C1)=O C1(CC(=O)N(CC(O)CN(C)C(c2coc(C(F)F)c2)=O)C)C=CS(=O)(=O)C1 C1(C(=O)NCCC(C)NC(=O)CCc2csc(Br)c2)NC(=O)OC1C N1(C(C(Br)=C(C)C)=O)CCCCC(C2CN(C(=O)C(C)(C)CN(C)C)C2)C1 n1(CC)ccc(C(=O)OC2C(CC(=O)NCC)CN(C(=O)CSCC)C2)cc1=O N1(C(CCN(CCCCC)C)=O)CCC(C#N)(C2(C#C)CCCC2)CC1 Cn1ncc2c1CN(C(c1cc3c(s1)CCC(C(=O)O)C3)=O)C2C(=O)O c1(C(N2C(CNC(CCC)=O)CC2)=O)c(Cl)sc2nnsc12 N1(C(C2C3CC=CCC23)C(=O)NCCOCC)CCP(C)(=O)CC1 C(=O)(C1CCc2ccccc21)N(C)CC1CC(F)CN1C(=O)COc1ccsn1 C(c1cc(C)cc(C)c1)=CC(=O)NCC1(O)CN(C(COCCC#C)=O)C1 C1(CNCc2c(C3CC3)cc(F)cc2Cl)COCC2(CCNC2)O1 C(=O)(C1=C(C#N)CCC1)NC1C(CC=O)CCCC1.CC(CCOC)N1CCC1 c1(OC)c(C(=O)NCC2CCCN2C(c2nnc(C)s2)=O)oc2ccccc12 N1(C(C(=O)NC(=O)NCC(N2CCCCC2)C)=O)CCN(CCCCF)CC1 c1(C(N2C(CNC(C(C)CO)=O)CC2)=O)ccnc(Oc2ccccc2F)c1 c1(N2CCC(N(C(=O)CCCCCF)CCC)C2)ncn(C)c(=O)c1Br c1(C(=O)NC2CCC3(C(NC(=O)C=C4CCC4)C3)CC2)coc2c1C(=O)NCC2 c1(C(N2C(CN(C(=O)CNC(=O)C(C)(C)C)C)CCC2)=O)ccc(N)cc1F C1(CNC(c2n(C=C)ncc2)=O)CCCCN(C(C2(CC(F)F)CCC2)=O)C1 N1(C(c2c(C(C)C)scn2)=O)CCCCC(NC(=O)C(C)N(C)C)C1 C1(NC(C2C(C)CCN2C(c2nc[nH]n2)=O)=O)CCCC(O)C1O C12(CNC(C(CCC)OC)=O)CCC(C1)N(C(=O)C(C1CC(F)(F)C1)O)C2 Cc1ccn2c(N(C(C3C(F)(F)C34CCC4)C(=O)NC3CCCC3)C)cnc2c1 C#CC1(C(=O)NC(C2CCCC2)CNC(=O)CC2CCC(=O)N2)CCC1 CCCCC(O)CC(=O)NCC1(Nc2ncc(C(=O)OC)cc2Cl)COC1 C(N=c1nc(N2CCC(SC(C)C)C2)c2c([nH]1)CCS2)C1(COC)CCC1 N(C(=NCC(C(F)(F)F)OC(C)C)NCC1CCCCC1)Cc1c(C)ccc(C)n1 c1(C(=O)NC2C=CC(CNC(C=CC(CC)=CC)=O)C2)nc(C)ccc1C C1(NC(C2C(C)C2C)=O)CS(=O)(=O)CC1NC(c1ncc(F)cc1N)=O C1(C(=O)NCC2COC(=O)N2)CC=CCN1C(C1CC1C1CC1)=O Cc1nc(NCCC2COCC(C)O2)cc(=NC2CC=CCC2)[nH]1 C1(CNC(C(C)(C)SC)=O)CC2(CCN(C(C3Cc4nncn4C3)=O)CC2)CO1 c1(OC)cc(C)sc1C(=O)NCC1CCCC1NC(=O)C=CSC Cc1ccc2cc(C(=O)NCC(C)NC(c3cc4ccsc4[nH]3)=O)ccc2c1 N1(C(CCn2ncc(C)c2)=O)CCC2(CCC(NC(=O)C(C)S(N)(=O)=O)C2)CC1 c1(C(=O)NCC2CC(NC(=O)C=C(Cl)Cl)C2)cncc(OC(F)(F)F)c1 N1(C(c2c(C)noc2)=O)CC2CCC1C1CN(C(=O)CSCC(N)=O)CC21 C(=O)(C1=C(Cl)CC1)NCCN(C(C(n1ccc(C)n1)C)=O)CC1CC1 N1(C(CC2CC(CC)C2)=O)CCCC2(NC(c3cnccc3C(F)F)=O)CC2C1 c1(C(=O)NCCN(C(c2c(CCC)nns2)=O)C)cccn2cc(C)nc12 c1(CC(=O)NCC(c2cccc(Cl)c2)OC)cn(C)nc1I c1(NC(C2C(CNC(C=C(C)C(F)F)=O)CC2)=O)ccc(OCF)cc1 C1(C(=O)NC2(CNC(c3cn(C)nc3O)=O)CC(OC)C2)CCCC12CCC2 n1(CC(=O)NCC(C(C)C)(C)NC(C2CCC(F)(F)CC2)=O)ccc(O)nc1=O C=CC1(C(=O)NC2(C)CCCC2(C)C)CCN(C(c2nccnc2OC)=O)C1 N1(C(C(C)CO)=O)CCC(C(=O)NC(C)CC(F)(F)F)CC1(C)C N1(C(C(CC)OC)=O)CC2CCC2(CCNC(=O)CC23COC(CF)(C2)C3)C1 c1(CC)ccc(C(=O)CCC(=O)NCCCNC(C2CCCC(O)C2)=O)cc1 CCC(C)C(C(=O)NC1CC2CCC1O2)N(C)C(c1nocc1C(C)C)=O c1(NC(C(CC(C)C)c2ccccn2)=O)nc(Cl)nc2cc(Br)cnc12 C1(CNC(c2ccn(C)c2)=O)CCCCN(C(=O)Cc2cccnc2N)C1 CC1CN(C(c2cc(C(F)F)nn2C)=O)CC(C)C1NCc1cc(C2CC2)no1 C(=O)(C(C(C)C)c1cccc(Cl)c1)NCCC1(OC)CN(C(C2CC2(C)C)=O)C1 CCCCCCCCC(=O)NCC1(C)CCCN(C(c2cnccc2CC)=O)C1 Cc1ncnc(C(=O)NCc2ccc(C(=O)NCc3cccnc3F)cn2)c1C CC(C)C(C)C(=O)NC1CN(C(c2csc(C(F)F)n2)=O)CC1C N1(C(CCCCC#C)=O)CCC2CCN(C(c3cc(Br)ccc3C)=O)CC12 Cc1c(C(N2CCCC(O)(CNC(C3CC34CC4)=O)C2)=O)ccc(Cl)c1Cl Cc1cc(O)ncc1C(N1CCCC(C(=O)NCCOc2ccncc2)C1)=O C1(C(=O)NCCC(C)NC(=O)COc2ccccc2)C2CCC12c1ccccc1 CC1CC(NC(=O)CC2CCCCC2)CN(C(c2ccnc(C(F)(F)F)c2)=O)C1 N1(c2nnc(COCC)n2CCc2cccc(C)c2)CCn2nccc2C1 C1(C(=O)NCCOC(C)=O)(NC(CCC)=O)CC1(C)C C(C)(CCCC(=O)NC(c1ccnn1CC)C)OC(C(=O)NCC)OCC Cc1nn(C)c(=O)c(C(=O)NCC(C(C)C(C)C)NC(c2ccc(Cl)[nH]2)=O)c1C c1(C(=O)NC(COCC)C)cncc(CNC(C2CC23CC3)=O)c1 c1(C(C(=O)CCCC(F)(F)F)=O)cnn2ccc(O)nc12.C12C3CCN(C13)C2=O C(C(C)(C(=O)NCCN1CCOCC1)NC(=O)Cn1ccnc1C)SC CN1CCC(C(=O)NC2CC(NC(=O)C=Cc3cscn3)C2)C1 C#CCC(CC(F)F)C(=O)NCC1C2CN(C(c3nccn3C)=O)CC12 c1(C(N2CC(NC(c3ccc(O)nc3)=O)C(F)C2)=O)cc2nccnc2cc1F c1(OCC(=O)N(C)CCN(C)C(C2CC2CC(C)(C)C)=O)cccc([N+](=O)[O-])c1 c1(C(=O)OCC)cnc(N(C)Cc2nc(Cl)cs2)c(C#N)c1 C12(CC(=O)NC(CN(C(C(C=C)C)=O)C)C)CCC(CC1)C2(C)C c1(C(N2CC(NC(COCC(C)(C)C)=O)C2)=O)cc(F)c(F)cc1Cl C1(C#N)(CC(=O)NCC2N(C(C(c3n(C)cnc3)O)=O)CC2)CCS(=O)(=O)CC1 C(=O)(CCCN(C)N=O)NC1(COC)CCN(C(C2CC(C#C)(O)C2)=O)C1 c1(NCCCNC(C2CCCCCC2)CC)ccnc(C)n1 C12CCCN(C1)CCO2.N1CCCC1Cc1cn(C(=O)NC2CC2(Cl)Cl)nn1.CO c1(C(C)C)ccc(S(=O)(=O)NC2CCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 C12(CNC(=O)C=Cc3ccco3)CCCCC1CN(C(c1cnsn1)=O)C2 n1(CCCC(=O)NCC2(F)CC(NC(C3C(C)(C)C3(C)C)=O)C2)c(O)nnc1O C(=O)(C(CO)NC(=O)C(N)=O)N(c1cccnc1)C c1(OC(c2nc(CS(C)(=O)=O)nn2-c2nc(C)nn2C)C)cccc(C#N)c1 c1(C(=O)NCC(C(C)C)NC(CCCOC)=O)cnc(CC2CC2)nc1O c1(C(N(C2CCN(C(=O)CCc3nncs3)C2)C)=O)cncc2nnn(C)c12 c1(OC)cc(C(c2nnnn2CC(F)F)NC2CCCC2)cc(Cl)c1 C1(NC(CC2(C)CCCO2)=O)C2CC(O)C1N(C(=O)Cn1nc(Cl)ccc1=O)C2 C12(C(=O)OC)CC(CO1)N(C(C1(NC(c3ccccc3CC(C)C)=O)CC1)=O)C2 C(CO)(C(=O)NCC1CCCN1C(=O)COC1CCCCC1)NC(C)=O.C1CN1 C(=O)(CC1=CCOCC1)NCC(C(C)C)C(=O)Nc1ccc(F)cc1 CC(C)CS(=O)(=O)CC(=O)NCCSCC(=O)Nc1ccc(=O)n(CCF)n1 C(=O)(C(CSC)C(C)C)NC12CCC(CNC(c3c(OC)noc3C)=O)(OC1)C2 C1(C(N2CCC(O)(C(C)NC(C3CC(F)C3)=O)C2)=O)CCc2ccnn2C1 C1(C(=O)OC)CCC(C)N(C(=O)NCc2nnc(-c3nc(Cl)ccc3Br)o2)C1 C1(NC(C(CCNC(C23OCCC(C)(C2)C3)=O)O)=O)CCCCC12CCC2 c1(-c2ncc(CN(CC(=O)OC)C(=O)C=Cc3nccs3)s2)ccccc1Br C(C(C(=O)NCC1(CNC(c2cnc(C3CC3)s2)=O)CCC1)C(N)=O)N(C)C c1(C(CC)NCC2(n3cncn3)CNC2)nc(Br)ccc1C N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CC2CC1C2NC(=O)COc1ccccc1 C(=O)(C(CC(C)C)N(C)C)NC(CC)CN(C(c1cncc(OC)n1)=O)CC C=C1CON(C(=O)CC2CCCCN(C(=O)CCOCC(C)C)C2)C(C)C1 CN(C)S(C)(=O)=NC(=O)NC1CC(c2ccc(Cl)c(F)c2)(O)C1 C12CC3CCC(C1)N3CC(=O)N2.c1(CC(=O)NC2CC2)c[nH]c(C(N2CCCC2)=O)c1 C(=O)(CC(CC)C(F)F)N1CCC(OC2CCN(C(CCOCCC)=O)CC2)C1 C(CC(C)(C)C)(C(=O)NC1CCN(C(c2ccc(F)cc2C)=O)CC1)NC(C)=O Cc1nnc(CCC(=O)NC(CO)C(C)NC(=O)CC2CC2(C)C)n1C C1(CNC(C2N(C)CCC2)=O)CC2COCC2N1C(c1csnn1)=O Cn1cccc1C=CC(=O)NC1CC(CNC(C2CC(=C3CC3)C2)=O)C1 c1(C(N2C3CN(C(=O)Cc4ccccc4Cl)CC32)=O)ccc2nc[nH]c2c1 CC1=CN=C2C=CC=CC12NCc1c(O)cnc2ccccc12 Cc1cc(C(=O)NCC(CO)NC(=O)CNC(=O)Nc2ccccc2)sc1Cl Cc1cccc(Br)c1OCC(=O)NC(CNC(C1(C)CC1)=O)CC(C)C c1(C(N2C(CNC(C=CS(C)=O)=O)CC(O)C2)=O)cccc(Br)c1F Cc1ccc(F)c(S(=O)(=O)NCCC(=O)NC(C)C(=O)OCC)c1.C(C)C S(=O)(=O)(CCC(C)C(F)F)Nc1ccc(Oc2ccc(C)cc2)cc1.C1C(=O)O1 C1(C#N)(OC)CC(C(=O)NOCC(=O)NCc2cc(C)c(CO)o2)C1 S(=O)(=O)(c1ccc(NCC2CCCSC2)cc1Br)NC(C1CCCO1)COC c1(C(C)C)ncc2c(n1)CCN(c1cc(NCCCc3nc[nH]n3)ncn1)C2 C1(C)(CNC(C(CSC)NC(c2ccc(C(C)=O)o2)=O)=O)CC=CCC1 C(CC(C(=O)NCCC(O)C1CC1)NC(c1cnc(S)nc1)=O)OC N1(C(c2c(C)non2)=O)CCN(C(C2C3CCCOC23)=O)CC(C)C1 c1(NCCOCCN(C(C2C(C)CC(C)O2)=O)C)c([N+](=O)[O-])cccc1[N+](=O)[O-] c1(N2CCCC(C(=O)NC)C2)nc2ncn(CC)c2c(=NC(C)c2nncs2)[nH]1 N1(C(C(C)(C)CF)=O)CCC=C(C(=O)N(C2CC2)CC2CCOC2)C1 C(=O)(C(CNC(=O)C(F)=C(C)C)CC1CC1)N(C1(COC)CC1)C C(=O)(CC(C)CC(F)(F)F)NC1C2(CN(C(c3c(CC)cccc3)=O)C2)CCC1 C#Cc1cccc(C(=O)NC2CC(C)(NC(c3cc(C)nc(C)c3)=O)C2)c1C N1(CCOC)CC(NC(=O)NCC2CCC(C(C)(C)C)O2)CCC1=O c1(OC)ccccc1CC(C)CC(=O)NC(CNC(=O)CCNS(C)(=O)=O)C1CC1 c1(CN2CCN(C(c3cc(NC(N)=O)ncc3)=O)CC2)c(F)cc(Cl)cc1F c1(C(=O)NC2C(CNC(C(C(C)C)SC)=O)CCC2)ccc2oc(S)nc2c1 C(=O)(C(CC(N)=O)NC(=O)CC1CCCOC1)NC1CCC(CC(=O)OC)C1 N1(C(CC2C(C)OC(C)C2)=O)CCCC2CN(C(=O)CCCC(F)(F)CO)CC12 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCCCCNC(=O)CCCCC1CC1)C S(=O)(=O)(c1cccc2c(Cl)nccc12)N1C2CCN(C(CC)=O)CC2CC1 C1(NC(C(n2cc(C(C)NC(c3ncccc3Cl)=O)nn2)C)=O)CC2CCC1O2 c1(C(=O)NC2(C(N(C)Cc3nc(C)on3)=O)CC2(C)C)cccnc1S c1(C(N(CC(CN(C(=O)Cn2cnnn2)C)O)C)=O)ccc(CO)s1 c1(C(=O)NC2(C)CC(NC(c3ccncc3)=O)C2)cccc(Cc2nc[nH]n2)c1 C(CCN(C)C(C1CCCCC1C(F)(F)F)=O)(C(C)C)NC(c1cc(C)[nH]n1)=O N1(C(C(COC)(F)F)=O)CCC(C)(C)C(CNC(C2(CF)CC2)=O)C1 c1(SCCNC(CCC)C2CC2(C)C)cc(Cl)ccc1Cl C(=O)(C(F)C(F)(F)F)NC(c1nc(C(F)(F)F)nn1C)C(=O)OC N1(C(C2(CC=C)CCC2)=O)CCCC(NC(=O)CC(CC)C2CC2)C1 c1(SCCC(=O)N(C)CCNC(C2CCCC2n2cccc2)=O)cccc(Cl)c1 Cc1ccc(CC(N2CCOCC2CCNC(C2(C(F)(F)F)CC2)=O)=O)c(Cl)n1 C1(C)(C(N2CCC(CC)(NC(C3CC4CCC3CC4)=O)CC2)=O)CCOC(C)C1 c1(C(=O)NC2C(OC)CN(C(c3cnn(C)c3Cl)=O)C2)cc2c([nH]1)CCOC2 CN=c1nc(N2CCC(c3nc[nH]n3)CC2)[nH]c(=NCC2CCCS2)[nH]1 N1(C(Cn2ncc(CC)c2)=O)CC2CCCC2(CNC(C2CC2OC)=O)C1 c1(C(=O)NC2(C)CC(NC(C(C)O)=O)C2)ccc(=N)[nH]c1 CCCCC(CNC(=O)CNc1cnn(-c2ccc(Br)cc2)c1)CCC C(=O)(CC1OC(C)(C)Oc2ccccc21)NCC(CNC(c1c(C)nc[nH]1)=O)C C(=O)(C1=CCS(=O)(=O)C1)NC12C(NC(C3CCN(C)C3)=O)CC(CC1)C2 N1(C(c2c(C)c(N)cnc2)=O)CCN(C(=O)C(c2ccnn2C)O)CC2(CC2)C1 N1(C(CC2C(C)OCC2)=O)CCc2nc(O)cc(C(=O)Nc3cccnc3F)c2C1 C(=O)(C1=CC2(CCN(C(=O)C=CC3CC3)C2)C1)Nc1ccc(C(C)C)nc1 C(C(C)(C)C(=O)NC(CC(=O)OC)C1CC1)NC(C(C=C)OC)=O C(=O)(C(O)C(C(C)C)NC(c1occc1C1CC1)=O)NCC1CN(C(C)=O)C1 O=S(=O)(NC1CCN(c2ccccc2F)C1)N1CCc2ccccc2C1 N1(C(c2cnc(COC)s2)=O)CCN(C(C23CC(F)(C2)C3)=O)C(CF)C1 N1(C(c2c(C)[nH]cc2)=O)CC2(COC(CNC(C3CCCC(O)C3)=O)C2)C1 C(C(C)C(C)(C)C)N(C(c1ccccn1)C)Cc1ccc(OC)o1 c1(C(=O)NCC2CN(C(C34CCC(CC3)O4)=O)CCCO2)ccc2nc[nH]c2c1 C1(C(=O)NC(CC)(C)CO)C=CCN(C(=O)C(=C2CCCCC2)F)C1 C(C(=O)N1CCOC(CN(C)C(c2cnoc2C(C)C)=O)C1)(C(C)C)SCC CC1COCCC1N(C)C(C1CSCCN1C(=O)CN1CCC(O)CC1)=O c1(C(=O)NCC2(C)CCN(C(=O)Nc3cc(F)ccc3F)C2)ccc(O)cc1Cl C(=O)(CC1=CCCCC1)N(C(C)C)CCNC(c1cocc1C(N)=O)=O c1(C(N(C2CCN(C(c3cc(Cl)c(Br)c(Cl)c3)=O)C2)C)=O)ccc2c(c1)OCO2 N1(C(C(C)=C(CC)C)=O)CCCOC(CNC(=O)CC2CCN(CCF)CC2)C1 C1(=O)CCCCN1.c1(C2CCN(CC)C2)ccccc1F.N12CCCC1C2=O c1(C(N2CC(CNC(c3ccoc3Cl)=O)C2)=O)cc2ccc(F)cc2nc1O NC1CC2CCC1CC2NC(c1c[nH]c(=S)cn1)=O Cc1ccc(NC(C2CCCCC2NC(=O)CCc2cnn[nH]2)=O)cc1CO N1(C(C(CC=C)C(C)C)=O)CC2(C1)CN(C(=O)COCc1ccccc1)CCO2 N1(C(C2(C#N)CC2)=O)CC(C2CCCN(C(=O)CC3CCC(=O)NC3=O)C2)C1 C(=O)(CCC(C)(C)C#N)NCCCN(CCCNC(c1ccon1)=O)C C(C(=O)NCc1cc(Cl)ccn1)(C(C)O)NC(C(C=CC)O)=O C1(NC(CC=C=C)=O)(CNC(=O)C(C)(C)CN2CCN(C)CC2)CCCCC1C N1(C(Cc2c(C)cccn2)=O)CC2CN(Cc3cc(Br)ccc3[N+](=O)[O-])CC2C1 C(CC(O)CNC(=O)CCOCCN(C)C(c1ccc(SC)o1)=O)OC Cn1c(C(N2CC3CC2CN3Cc2c(Cl)cncc2Cl)=O)cccc1=O Cc1c(C(=O)N(C)CC2CCCCN2C(=O)C(C)(C)F)cnn1CCO N1(C(C2C(COC)CC2)=O)CCC2(CCCN(C(=O)CSc3cccnc3)C2)C1 C#CC1CN(C(c2cc3ccsc3s2)=O)CCN1C(=O)C(F)CC1CCOC1 CC1(C(=O)NCC2CN(C(=O)CCOC3COC3)CCO2)CC2CCC1C2 Cc1cc(C(=O)NC(CNC(C2CC23CC(F)(F)C3)=O)CC(C)C)c(Cl)cc1N c1(NCCc2nc(C(F)(F)F)sc2)nc(N2CC3COCC3C2)nc2sccc12 CCC(C)CCCC(=O)N(CC(=O)NCCO)C(c1cn(CC)nc1C)=O c1(C(=O)NCC2CCN(C(CC(C)F)=O)CC2)ccc2c(c1)C(=O)CCC2(C)C C12(CNC(COCC(=O)OC)=O)CCCC1CN(C(C1(C)COCCO1)=O)C2 N1(C(C2C(CCC)CCC2)=O)CC(F)(F)CC1(C)CNC(c1snnc1C)=O C(=O)(C(=O)N1CCC(O)CO1)OCC(C)OCC1CC1 c1(N(C(C)C(=O)NCC(C2CCC2)NC(C2CC2)=O)C)cc2sccc2cn1 C1(N(C(C2CCC(OC)C2)=O)C)CC2CCC(C1)N2C(=O)C(C)(C)C1CC1 c1(NC(C=CC(=O)NCC(c2c(C)cc(F)cc2)(F)F)=O)nc2ccccc2[nH]1 n1(C(C)C)ncc(Cl)c1C(N1CCC(CCN(C)C(C2(C#N)CC2)=O)CC1)=O c1(C(=O)NC2CC(CNC(CC(CC)C3CC3)=O)OCC2)nc2ncccn2n1 C1(CC)C(NC(=O)CN(C)S(N)(=O)=O)CCN1C(c1cn(C2COC2)nn1)=O C1(CC=C)(C(=O)NCC(C)(O)C2CC2)CN(C(=O)C(F)OC(F)(F)F)C1 c1(C(=O)NC2CN(Cc3ccc(OC)s3)CC2O)cnc2ccccn12 c1(OC2C(C(=O)Nc3ccc(Cl)cc3)CCC2)ccc(Cc2nnsn2)cc1 N1(C(C(CC)(C)O)=O)CCC(NC(=O)C(C)(C)CCOC)C(CO)CC1 N1(c2nc(NCCC(=C)C)c3c(n2)scc3)CCc2c(Cl)cc(Br)cc2C1 Cc1coc(C(=O)NCC2CC(NC(=O)C(c3cnn(C)c3)C)C2)c1C C1(CC(=O)NCc2ccc(C)s2)CC(NC(c2cc(O)nn2C)=O)C1(C)C C(=O)(C1=NOC(C)(C)C1)NC(CN(C(c1scnc1Br)=O)CC)C C12(NC(Cc3cccc(C)c3)=O)CCCC1N(C(c1ccc(F)cc1Cl)=O)CC2 c1(CC(C)C)ccc(C(=O)NC2C=CC(N)C2)cc1.c12ccc(nc1)n2CCO c1(C(=O)OC)c[nH]c(=NCC(C)CNC(C2CC(C3CC3)C2)=O)s1 c1(C(=O)NCC(CO)NC(C=CSC)=O)cnn(C)c1C(C)(F)F C1(C(N(C)CC2(CNC(C3CCC(=O)N3)=O)CC2)=O)CNS(=O)(=O)C1 C1(CC(=O)NCCCC(O)CO)CC2(C1)CN(C(C1(F)CCOC1)=O)C2 c1(C(=O)NC2C(NC(c3nc(C(=O)OC)oc3)=O)CCCC2)c(C)[nH]c(C)c1C c1(C(=O)NC(C)CCNC(C2CC(=O)N(C3CC3)C2)=O)cccc(Cl)c1F Cc1nc(NCC23CC(CN2C(c2ns[nH]c2=O)=O)C3)cc(O)n1 c1(C(N2CCC(NC(=O)CCC3OCCO3)(CO)C2)=O)ccn2c(O)nnc2c1 c1(C(C)NC2CCCC2O)ccc(NC(=O)C2CC2)cc1 Cc1cccc2oc(C(N3CC(NC(=O)CCc4ccoc4)C4(CC4)C3)=O)cc12 C1(C(=O)NC(CCNC(C(C=C)OC)=O)(C)c2nnnn2C)CCOC1C=C C1(CC(=O)NCC2CN(C(CC(=O)NCC)=O)CC2O)CCC(C)(C)CO1 CCCCC(C(=O)N(C1CN(C(=O)C=CC2CC2)CC1O)C)N(C)C c1(N(C)CC2(N(C)C)CCC2)nc(N2CC3C(C(F)(F)F)C3C2)c2ncsc2n1 c1(CN(C(C(=O)NCCC)CCSC)CC(F)F)ncc(C)cc1OC c1(CC(=O)OC)cccc(NC(=O)CCNC(=O)NC(C)CN2CCCC2)c1 C1(C(=O)NC2CC(N(C(C(C)Cc3cnco3)=O)C)C2)CC12CCCCC2 N1(c2nccc(-c3ccccc3)n2)CC(O)CC2(CC2)C1 C1(C(=O)Nc2ccc(N3CCC(O)C3)cc2)C2CC3C1C3C2F c1(C(=O)NC2(C(C)NC(CNC(C(C)C)=O)=O)CC2)nc(-c2cc[nH]n2)cs1 c1(C(=O)NCCC2OCCCN(C(C3COC(=O)O3)=O)C2)n[nH]c2cccnc12 NC1CS(=O)(=O)C2CN(C(=O)CCc3c(F)cc(F)cc3Br)CC12.C(C(=O)O)N C#CC1(NC(=O)C(C)(C)CN(C)C(c2cc(C)nc(C)n2)=O)CCCCCC1 C1(NC(C2N(C(c3nc(C)sc3)=O)CC=C2)=O)CCCC2(CC1)CC2 c1(SC)ccnc(N2CCC(NC(c3ccnc(O)c3)=O)C2)n1 C(=O)(C(O)C(C(C)C)OC)NCC1(C)CCCN(C(c2ccc(C#C)cc2)=O)C1 N1(C(CNC(=O)Nc2c(C)cccc2)=O)CCN(C(=O)C(C)(C)N(C)C)CC(O)C1 c1(C(=O)NCC(CN(C(c2cccc[n+]2[O-])=O)CC)(C)C)cn2nc(C)sc2n1 Cn1cncc1C#CC(=O)Nc1cccc(-n2cncn2)c1 N1(C(C2(C)COCCO2)=O)CCC2CN(C(c3ccc(F)cc3C(F)F)=O)CC12 CCC(N=c1[nH]c2cc(Cl)ccc2n2cncc12)c1cccc(C)n1 C1(CC(=O)NCCOCCN(CC=C)C)CCC(=O)N1 C1(CNC(c2c(C)n(-c3ccccc3)nc2)=O)CCN(C(=O)C(N)=O)C12CCC2 c1(OC)ccc(O)cc1-c1csc(NC(=O)CSCc2cccs2)n1 CC1(C)CC(C(=O)NCC2(NC(c3ccc(N4CCCCC4)cc3)=O)CC2)CO1 N1(C(=O)Cc2nncs2)CC2(C1)CN(C(C1CN(C3CCCCC3)C1)=O)CCO2 C12CCC(CC1)COCC(=O)N2.Cc1cscc1C(=O)N(C1CCOC1)C1CC1 C1(NC(c2c(C)cc[nH]2)=O)CCCC(NC(C2(CC(C)C)CCCC2)=O)CC1 C1(NC(CCS(=O)(=O)NC)=O)CCC2(CCCN(C(c3cc(OC)n[nH]3)=O)C2)C1 C(=O)(C#CC1(C(F)(F)F)CC1)NC(C)C(CO)NC(=O)C(C)(C)C(F)F C(c1ccccc1)=CCC(N1CC=CC(C(=O)NCCc2ccncn2)C1)=O c1(C(N2C(CNC(C(=O)N(C)C)=O)C(C3CC3)CC2)=O)cccc2nsnc12 c1(CC(N2CC(O)CC(NC(C3(N=[N+]=[N-])CC3)=O)C2)=O)ccc2c(c1)CCOC2 c1(C(=O)NC2CC(O)(CNC(c3c(C)n(C)cn3)=O)C2)ccc(O)nc1Cl c1(C(N2CC(F)CC(C(=O)NC(C#C)C)C2)=O)cc(O)cc([N+](=O)[O-])c1 c1(C(=O)NC2C(CNC(c3ccnnc3)=O)CC2)nc2ccc(Br)cn2n1 C1(C(=O)NCc2c(C)ccc(F)c2)CC12CCN(C(=O)C=Cc1ccsc1)CC2 C(C(C(F)(F)F)N1CCN(C(C2CCCCS2)=O)CC1)NC(COC)=O c1(C(=O)NCC(C)(CO)NC(c2ccc(C#C)cn2)=O)cccc2c1CCC2 C1(CNC(C2CCC2)=O)CCC2(CCN(C(c3cnc4n3CCS4)=O)CC2)CO1 N1(C(c2c(OC)ccnc2F)=O)CCCN(C(=O)C(C)(C)OC(C)=O)C(C)C1 C1(C)(C(N2CC(C(=O)NC(C)Cn3cncn3)(CC)C2)=O)CCCC1O N1(C(c2c(C)cns2)=O)CCC(C)(CNC(c2ccc(O)c(N)c2)=O)CC1 c1(C(=O)NCCC(CNC(C2(CC)COC2)=O)O)[nH]cnc1C#N N1(S(=O)(=O)c2ccc(O)cc2)CCc2cc(-c3ccc4nonc4c3)cnc2C1 c1(C(N2CC(CN(C(C(CC)(C)CC)=O)C)OCC2)=O)cnn2ccn(C)c12 C1(CNC(c2ccnc(OC)n2)=O)(CO)CC12CCN(C(C1(O)CCC1)=O)CC2 N1(C(CC(=O)N(C)C)=O)CCCCC(C2CN(C(C34CCCC3C4(F)F)=O)C2)C1 CC(C)(C)C1=NOC(C(=O)NCCCNC(=O)CCCN2CCCC2)C1 C1(C(=O)NC2(C)CCOC2=O)(CC)CCN(C(C2CN(C)CCO2)=O)CC1 CCC(CN(C)C)C(=O)N1CC(C)(NC(=O)Cc2csc(Br)n2)C1 c1(C(=O)NC2CC(NC(C(C)=CC3CC3)=O)C2)cccc(Br)c1Br CCCCC(C)(F)C(=O)NCCCC1(N(C2(CC(=O)NC)CCC2)C2CC2)CC1 CC1CCC(F)(C(N2CCN(C(c3sccc3F)=O)C(CC3CC3)C2)=O)CC1 C#CCC(C)(CNC(C1CC2(CC2)CN1C(=O)C(O)C1CCCC1)=O)CO N1(Cc2nnn(C)n2)CCCCC1CNC(=O)CCNC(=O)Cc1ccsc1 c1(CNC(C(n2cc(CCc3ccccc3)nn2)C)=O)ccn(C)c1 c1(C(N2CC3CN(C(=O)C(Cl)(Cl)Cl)C3C2)=O)cc(I)c(F)cc1F N1(C(C(CCOCC)NC(c2cnc3n2CCC3)=O)=O)CCC(C)C2(CCC2)C1 C1(C(c2ccco2)C)CCCN1C(=O)NCc1c[nH]nc1C1CCC1 c1(C(N2C(C)CC2C(N2CC(F)(F)C2C2CC2)=O)=O)cn2ccccc2n1 C1(NC(c2ccoc2C(F)(F)F)=O)CN(C(c2cocn2)=O)CC12CCC2 c1(N2CC(OC)(CNC(c3ccc(C(C)C)nc3)=O)C2)nc2cccc(F)c2o1 c1(C(N2CCN(C(C(CC=C)CC)=O)C(C3CC3)C2)=O)ccc(C)c(F)c1F N#Cc1ccc(Br)cc1C(N1CC2CC2(C(=O)Nc2ccnc(Br)c2)C1)=O c1(C(=O)NC(C2N(C(C3CC(=C)C3)=O)CCCC2)C)cnc2nc(C)oc2c1 c1(CC(=O)NC2CCC(CNC(CC(C)C)=O)C2)cnn2ccccc12 c1(OCC(=O)NCC2CN(C(CC(=O)OC)=O)CC2F)cc(Cl)c(Cl)cc1Cl Cc1cncc(CC(=O)NC(C)CCNC(c2onc(C)c2C)=O)c1 C=C1CCN(C(=O)COCC2CC2)C(C(N2CC(c3nocc3C)C2)=O)C1 C(=O)(C1=NN(CC(=O)O)C(=O)CC1)Nc1ccc(OCCOC)nc1 C1(CNC(c2ccc(C)o2)=O)CCC(C)(C)CN1C(=O)CCCCc1cnc[nH]1 CC1OOC(=O)NC1C(N1CC(CNC(c2cc(C3CC3)no2)=O)C1)=O C1(C)(COC)C=CCN1C(=O)CC(CNC(c1ccnc(CO)c1)=O)C1CCC1 C1(NC(c2nnn(CC)c2C)=O)(CNC(c2csc(Cl)c2)=O)CCCCC1C CCC(C)CCCC(=O)NCC1CC(NC(=O)CCOc2ccc(Cl)cc2Cl)C1 C1(CCCC)CN(C(c2sc(OC)nc2Cl)=O)CCN1C(=O)C(C)c1cccs1 CC1(C)CN(C(C2(O)COC2)=O)CC2(CN(C(=O)C=C3CC3)C2)O1 N1(C(C(CCCCC)O)=O)CC2CCCN(C(c3ccc(O)c(F)c3F)=O)C2C1 c1(CC)cncc(CNC(=O)CN(CC(C)C)C(C23CCCC2C3)=O)c1 c1(OC)ncc(C(N2CCC(NC(c3cscc3C)=O)C23CC3)=O)nc1C c12ccc(Cl)cc1S(=O)(=O)NC2=O.c1(NS(C)(=O)=O)nc2ccccn2c1Cl c1(N(C(c2cc(Br)c(F)cc2Br)=O)CC2(C)CNC2)ncc2cccc(Br)c2n1 C1(CC(=O)NCC(C)(CO)NC(CCCC(C)C)=O)CCc2sccc2C1=O c1(C(N(C2CN(C(c3ccnn3C)=O)CC2(C)C)C)=O)cc2c(=O)cc[nH]c2s1 c1(C(N2C(C3CCN(C(C=C(C)C)=O)C3)CCC2)=O)cnn(C(C)C)c1C C1(CC(=O)NCc2ccc(C(=O)NCC3CCCCC3)nc2)CC(=O)NC1=O c1(N(C)CC2N(C(CCC3C(C)=NOC3=O)=O)CCC2)nc2cccc(C)c2o1 C=CC(CC)CC(=O)N1CCC(N2CCCC2)C1.C1C(=O)NO1 CCCC(C)(C)C(=O)NC1CC(CCNC(c2ccnc(SC3CC3)c2)=O)C1 c1(C(N2CC(NC(C(C)(C)C3CC3)=O)C3C2C3)=O)ccc(C(F)F)c(Cl)c1 CCC(C)CCCCC(=O)NCCC(=O)NC(C)CC(C)(C)CO CCCCN=C(NCC1CC1CC)NC1CC(C#N)C1 c1(C(C(=O)OC)NC2C(C(=O)OC)CC2)ccc2c(c1)OC(C)(C)O2 C1(CCCN)(NC(C(CO)CCc2ccncc2)=O)CCCCC1 C1(C(C)NC(Cc2c(C)ccs2)=O)CCCN(C(=O)Cc2noc(C3CC3)n2)C1 CC1(C)C(C(=O)NCCCCCCO)CCN1C(c1ccccc1Cl)=O CC(CN1CCN(C)CC1)N=c1ccnc(C(=O)Cc2ccc([N+](=O)[O-])cc2)[nH]1 C=CCCCC(C(=O)Nc1cccnc1)NC(=O)CCNC(=O)CO CN1C(=O)CCC1CC(=O)NCc1ccc(CCNC(C2(C#N)CCC2)=O)cc1 c1(NC(N2CCCC(C(=O)NNc3ccccn3)(C)C2)=O)ccc(S(N)(=O)=O)cc1 N1(C(CCc2onc(CCC)n2)=O)CCCC(N(C)C(C2CC=CC2)=O)C1 C(=O)(CCCCCCC(C)C)N(CCN(C(c1c(C)nc(O)cc1)=O)C)C C(=O)(C(C)(C)C(C)(C)C)NCCOCCNC(C(C1CC(F)(F)C1)OC)=O c1(C(C)NC(=O)CC=CCNC(c2cccnc2O)=O)ccc(O)nc1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCC3)=O)C2)cnc2n1CCCC2 c1(OC(CC)Cc2ccc(N(C)C)cc2)ccc(Br)c(C(F)(F)F)c1 c1(OC)noc(C(N2CC(CNC(=O)Cc3n[nH]c(C)n3)C(C)C2)=O)c1Br c1(OCCC(=O)NC(CC)CNC(=O)CSCCC#N)cccc(C)c1 c1(CC)nc(=NC(=O)N2CCC(Cn3cc(CCCCO)nn3)C2)n(C)[nH]1 CC(C)CCC(=O)NC(C)(C)COCCCNC(c1cnn(C2CC2)c1Cl)=O n1(CCCC)ncc(C(=O)NC(CO)C(C)NC(C2(C)CCCOC2)=O)c1C c1(N2CCC(CC=C)C2)nc(N2CCC3(CC2)CCN3CC)nc2c(F)cccc12 c1(C(N2CC(CNC(CCCC#C)=O)C(C)C2)=O)cc(C#N)ccc1C C12(CNC(C(c3ccccc3)SC)=O)CN(C(=O)CCC3CC3)CC1CCO2 C=C(C)CN=C(NCC(c1ccc(F)c(Cl)c1)O)NCC(C)(C)C#N C1(NC(C(C)(C)SC)=O)CN(C(=O)COc2ccc(Cl)cc2C)CC1C1CC1 c1(OC)cccc2c1OCC2NC(c1ccc(CNCCO)cc1)=O C(=O)(CC1OCc2ccccc21)N(C1CN(C(C2CNC(=O)N2)=O)CC1(C)C)C C12(C(=O)NC(C)CCCNC(C3(N4CCCC4)CCC3)=O)CCCC1C2(F)F c1(C(=O)NC(CCN(C(C=C(C)Cl)=O)C)C(C)C)cnc(C2CC2)nc1O N1(C(C=CC=CC)=O)CCC(n2cc(CNC(=O)C(CC)N(C(C)=O)CCCC)nn2)C1 c1(N(C2CCNCC2(C)C)C(c2nccc(C)c2)=O)ncnc2cccnc12 C(=O)(CC(O)CN(C)C)N(C(CC(=O)N(CC(=O)OC)C)C)c1coc(C)n1 C(=O)(C#CC1CCOC1)NC1CC(C)(NC(=O)C(c2ccc(Cl)s2)=O)C1 CC1=NOC(CN2CCCC2)C1.C12COCC1CN(C)C(=O)C1CC(C1)NC2=O C(C)(C(=O)NC(C)CN(C)C(C)C)(C1CN(C(CC2C(CC)C2)=O)C1)OC c1(C(=O)NC2CC3(CC(CNC(C=COCC)=O)C3)C2)cc2ccccc2n1C C(C(=O)NC(C1CC(NC(c2cn(C)cn2)=O)C1)C)(C(C)C)OCC Cc1ccc(=O)n(CC(N2CCC(N(C(=O)C(C3CCCCC3)F)C)C2)=O)n1 C1(NC(c2ccnn2C(F)F)=O)CCN(C(C2CCC=CCC2)=O)CC1 c1(OC)c(F)cc(C(=O)NC2CN(C(C3(C)CCCC3)=O)CC2F)cc1F C(C(O)C(C)(C)O)NC(C1(CC)CN(C(=O)Cn2cccc2C(=O)O)C1)=O c1(OC)c(C(=O)NCC2CCN2C(=O)C(C(C)O)NC(C)=O)csc1C N1(Cc2c(C)nc(C)o2)CCC(F)C(Sc2ccccc2)C1 CC(C)CC(C)(O)C(=O)NC1CCN(C(c2c(O)cc(Br)cc2F)=O)CC1 c1(C(N2C(CN(C(C(CC)C)=O)C)CCC2)=O)cc(C)nc2ccc(F)cc12 c1(C(N2CCCC(NC(Cn3c(C)cnc3)=O)CC2)=O)nc[nH]c2ncnc1-2 Cc1nc(CNC(C2C(C)C2C)=O)oc1C(=O)NCCCN(C1CCCC1)C C1(C(=O)NCC2(CNC(C(C=C=C)C)=O)CCOCC2)CC2(CCOCC2)C1 c1(C(=O)NC2(CNC(C=C(CC)C)=O)CCOC2)cc(-c2ccncc2)ccn1 C1(O)(C(C(=O)NCCN(CCC)CCC2CCOC2)F)CCCC1 c1(OCC(=O)NCCCC(CO)NC(C2CCCSC2)=O)ccc(F)nc1 C1(CC(=O)N(CCCN(C(=O)C=C2CCC2)C)C)CC(=O)c2ccccc2C1 Cc1cc(O)ccc1C(=O)NC1CCC1NC(=O)CC1CC(C)C1 CCC(C)C(C(=O)NCCCCN(CCCNC(=O)C=Cc1cc[nH]n1)C)OC Cc1cc(=O)ccn1CC(=O)NC1CCCCC1NC(=O)C1=CCCOC1 C1(CC(N2CC(NC(C3CCN(C(=O)NC)CC3)=O)C2)=O)CCN(OC)CC1 C1(OC)CC(NC(C2(C)COC2)=O)CN(C(C)=O)C1.c1(C(=O)N)ccsc1 c1(CCC(=O)NCC2CC2CNC(C2CC2C(F)F)=O)ccc(F)c(F)c1 N1(C(CC(C)C(F)F)=O)CCC2(CCN(C(=O)CCC3CC3(Cl)Cl)CC2)C1 C1(CNC(C2N(C(N)=O)CCC2)=O)CC2CCC(C1)N2c1cc(F)ncn1 CC(Cc1cnn(C)c1)C(=O)NC(CNC(C1(C#N)CCC1)=O)C1CC1 CC1=C(C(=O)NCC2CCN(C(=O)C(C)(O)C3CCOCC3)C2)CCC1 N1(C(C(C)n2cnnn2)=O)CCC2(CC(NC(=O)CN3CCNC(=O)C3)C2)C1 N1(C(CN(C(=O)C(C)CC#N)CC(C)C)=O)CCC(O)(CO)C1 c1(N2CCCC(C(=O)NC)C2)nc(N2CCC3CC3C2)nc2c1COC2.C(C)(=O)N C=CCC(C)(C)CC(=O)NCC(C(=O)N(C1CC1C)C)OC C1(NC(C2CN(C)C2)=O)CCC(CNC(c2csc(-c3cn[nH]c3)n2)=O)C1 N1(C(C2CCC=CO2)=O)CCCC12CCN(C(C13CCCCC1C3)=O)CC2 C1(CCNC(C(CC)(C)OC)=O)CC(F)(F)CN1C(=O)C(COC)OC c1(CC)ccc(CCC(=O)NCC(CNC(C2C3CCN2CC3)=O)OC)cc1 N1(C(c2ccc(CO)c(F)c2)=O)CC2CCC1C(Nc1ncnc(Cl)c1Br)C2 c1(CCc2cnc(SCC(=O)Sc3ccc(C)cc3)s2)nc2ccccc2[nH]1 N1(C(=O)NCC2(SC)CCCC2)CCN(C(C)C)CC1 C(=O)(CC1COc2cc(O)ccc21)N1CC(NC(c2cnn3c2CCCN3)=O)C1 N1(C(=O)NCC(c2ccc(Cl)cc2)C2CC2)CCOC2CCCC12 c1(C(=O)NCC(CC)NC(=O)CNC(C)=O)oc(Br)nc1C c1(C(=O)NCC2N(CCCOC)CCC2)ccc2ccn(C)c2c1 c1(C(N(CCCNC(Cc2ncc(CC)[nH]2)=O)C(C)C)=O)ccc2ocnc2n1 C12(C(=O)NCCC3N(C(=O)C(c4ccc(Cl)s4)=O)CCSC3)CCC(CC1)CO2 CN1C(=O)OCC1C(=O)NCC(CC(=O)N1CCSCC1C1CC1)N(C)C c1(OCC)c(CC(=O)NCCN(C(=O)CC2(O)CCCC2)CC)cccc1Cl n1(C(C)C)cc2c(n1)C(C(=O)NCC1CCN(C(=O)CC3CCCC3)C1)CCC2 N1(C(CC(C)OC)=O)CCN(C(C2(Cc3ccc(O)cc3)CCOC2)=O)CC1 c1(C(N2CC(C(N)=O)CC(OC)C2)=O)c(F)cc(Br)c2c1OCO2 C(=O)(CC1=CCN(C)CC1)NC(C1CN(C(C2CCCCC2)=O)C1)C.CC=C(C)C C1(CN(C)C(c2cscn2)=O)C2CN(C(C3CCN(C)C3)=O)CC12 C1(C(=O)NC2CCCC(NC(c3ccncc3O)=O)C2)CC2CCC(C1)S2 c1(C2N(Cc3c(O)ccc(O)c3)CCC2)cccc2ccccc12 C1(CNC(C2CCCC(OC)C2)=O)CC(C)(C)CN1C(c1ccc(CO)cc1)=O C1(CC(N2C(CC(N)=O)CCC2)=O)CCCN(C(c2ccsn2)=O)C1 C(c1ccc(Cl)cc1F)=CC(=O)N(C(C)CCNC(c1n[nH]c2c1COC2)=O)C c1(C(=O)NCC(C)(C(C)C)NC(c2c(CC)cco2)=O)ccc(F)cc1F N1(C(C=CCCC)=O)CC(NC(=O)C(C)=C2CCCC2)CC2(CC2)C1 C12(C(=O)NCC(C)(C)NC(CCc3n(C)ncc3)=O)CC(C)(C1)OC2(C)C c1(COC)c(C(N2CC(OCCNC(C3CC=CC3)=O)C2)=O)sc2ccccc12 c1(C(=O)OC)ccc2c(c1)C(NC(=O)N(C)CCOc1ccccc1C)CC2 Cc1c(Br)ncc(F)c1NC(=O)CCC(c1ccc(F)c(F)c1)=O C(=O)(C1CCc2ccccc21)NC(CCOC)C(=O)N(c1sccc1C)C Cc1cccc(CN2CCN(CC(=O)NC(C3CCC3)C)CC2)c1O N1(C(C(C)SC)=O)CC(O)(CNC(c2cn(CCO)nn2)=O)C1 O(NC(=O)C1=CCN(C(C2CC=CC2)=O)C1)C(CC)CC N1(C(c2ccc(C)s2)=O)CC2CCCC2(NC(c2cccc(O)c2C)=O)C1 C1(NC(C(C)n2cccn2)=O)CC2CC(NC(c3cc(C(F)F)ncn3)=O)C1C2 c1(N(CCNC(C2(CCC)CC2)=O)C)nc(CC(C)(C)C)nc(=N)[nH]1 Cc1c(C(=O)NC(c2ccc(C(=O)O)cc2)C)cccc1[N+](=O)[O-] Cc1ccc(C)c(OCC(N2CC3(CCC3NC(C3CCCCS3)=O)C2)=O)c1 N1(C(c2cc(C)oc2C)=O)CC(NC(=O)CC2CC(C)(C)C2)C2(CC2)C1 C1(CNC(COCCC=C)=O)CC(NC(c2cc(C)ccc2F)=O)C12CCC2 N1(C(Cc2c(C)scc2)=O)CCOC(C(=O)NCCc2ccc(O)cc2)C1 c1(NC(C2CCCCN2Cc2ccccc2[N+](=O)[O-])=O)cc(F)c(F)cc1F c1(C(N(C2CCCC(NC(C3CCOCC3)=O)C2)C)=O)cnc2cccnc2c1 c1(NCC2(CCNC(=O)CC(F)(F)F)CC2)cc2cc(Br)ccc2[nH]1 C12(NC(C(CSC)OC)=O)COC(C1)C(NC(C1(CF)CCC1)=O)C2 C1(NC(C(CC)=CC)=O)CCCCCC1NC(=O)CCn1nc(C)nc1C N1(C(C(C)c2ccsc2)=O)Cc2ccccc2C1CNC(=O)C(F)OC(F)(F)F CCC(C(=O)N1CCC(CN(C(c2ccnc(CO)c2)=O)CC)CC1)C(C)C C1(OC)CN(C(=O)CCn2ccc(C)n2)CC1NC(=O)C=Cc1nccs1 c1(C(=O)NC(CCOC)C(=O)N(C)C(c2nc(C)no2)C)ccc(C)c(O)n1 C1(C(=O)NCCOC(CNC(c2c(C)n[nH]c2C)=O)(C)C)CC2(C1)CC(C)(C)C2 c1(C(c2n(CCCC)nnn2)OCC)cc(NCC(C)C#N)c(F)c(F)c1 c1(C(=O)NCC(CNC(C2C(C(N)=O)C2)=O)F)n[nH]c2ccc(F)cc12 Cc1nc(NC2CCCN(C(c3cccc(=O)n3O)=O)CC2)c(C)c(O)n1 N1(C(=O)C=C2CCC2)CC(=O)NC2CN(C(c3ccc(C4CC4)cc3)=O)CCC12 c1(NC(C2C(Nc3cc(C)ncn3)C2)=O)c(C)ccc2c[nH]nc12 Cc1ccc(F)c(C(N2CC(C(N3CCCC(CCO)C3)=O)OC(C)C2)=O)c1 N#Cc1cc(F)ccc1CN1CCC=C(C(=O)NC2COC3(CCCC3)O2)C1 C=CC1CCCN(C(=O)Cc2coc(-c3ccc(Br)cc3)n2)C1 Cc1noc2cc(C(N3CCCN(C(=O)CCC4CCCO4)C(C)C3)=O)ccc12 C1(C(=O)NC2CN(C(c3c(C)cns3)=O)C2)(CN(C)C)CCCCC1 N1(C(C(C(F)(F)F)OC(C)=O)=O)CCC2(CC1)CN(C(=O)CC(C)O)C2C(C)C C(C(C)(C)C1=CCCC1)NC(c1c(C)cn(C)n1)c1nnnn1C C1(C(N2CC(C)(OC)C2)=O)CCC(CNC(C2(C)CC=CCC2)=O)CC1 OC1CC2(CCN(c3ncc4c(n3)CCCC43CN3)CC2)CC1.COC c1(C(=O)OC(C)C)ccc(C(N2CCC(CNC(C3CC3(C)C)=O)C2)=O)cc1 c1(C(=O)NC2(CNC(CC3C(C)C3)=O)CCCC2)ccc(-n2cncn2)c(F)c1 CN1CCN(C(=O)N(Cc2ccccc2)Cc2ccoc2)C(c2cccc(F)c2)C1 CCC(C(=O)NC1(C)CC(C(=O)NC2(c3ccccc3Cl)CC2)C1)C(C)O C1(NC(=O)OC(C)(C)C)CCC(NC(c2cn(C3CCCC=C3Br)nn2)=O)CC1 C12(C(=O)OCC)COCC1CN(C(C1CCC(OC)C1)=O)C2.c12[nH]c(nc1C)C2 c1(CN(C2CCN(C(c3ncc(F)cn3)=O)C2)C)c[nH]c2c(Cl)cccc12 C(=O)(C1=CCCCCC1)N1CCC(O)(CCNC(C2CC3CC2C3)=O)CC1 c1(C(=O)N=c2[nH]nc(C(F)F)s2)nnc2ccc(-c3cnn(C(=O)NC)c3)cn12 c1(C(C)=O)ccc(CNC(c2ccncc2)C(=O)NCCCOC)cc1C N#Cc1cccc(CC(N2CC3CC3(NC(C3CC4CCC4C3)=O)C2)=O)c1 Cc1cc(C(=O)N(CCCNC(C2CCCCC2F)=O)C(C)C)cc(C)c1 CC1CN(C(C2CCCCN2C(c2ccc(Cc3cnc[nH]3)cc2)=O)=O)CCO1 c1(C(N2CCC(N(C(=O)CSC(F)F)C)C2)=O)cc(F)c(F)c(O)c1F c1(C(N2CCC(NC(C(CC)N3CCCC3=O)=O)C2C)=O)cc(C)cnc1Cl C1(C(=O)Nc2c(C)ccc(NCO)c2)CCN(C(=O)C(=O)C(C)C(C)(C)C)O1 C12(C(N3CC(C)(C(=O)OC)C3)=O)CC(CCO1)N(C(=O)CC1CCCSC1)C2 c1(C(N2CC(OCCNC(CN(C)C3CC3)=O)C2)=O)ccc(F)c(Cl)c1N C(C1CCc2ncnn21)N1CC(NC(C2(c3cc(C)no3)CCCC2)=O)C1 N1(C(C2(C(C)C)CC2)=O)CC(NC(C2CC2(C)C(F)F)=O)C(c2ccccc2)C1 CC(C)C(F)(F)CC(=O)N(C)CC1(O)CCN(C(C2(C)CC3CCC2C3)=O)CC1 c1(C(=O)NC2CCC(C(=O)NC3C(C)(COC)CCC3)C2)ncc2ccccn12 CC(C)CC(C)(CNC(=O)CCC(=O)N(C)C)OCCCNC(C1C2CCC12)=O C1(C(=O)NC2C3CN(C(c4c(CC)cno4)=O)CC2C3)CCc2ccccc2C1 O=C(C(F)(F)C(O)C1CC1)NCC1C2CN(c3ccc(Cl)nn3)CC12 Cc1cc(F)c(C(=O)NC2CC2CNC(C23CC4CC2C3C4O)=O)cc1F CCC(C)(CCNC(C1CCCO1)=O)NC(=O)CC(O)CN(C)C C1(C(=O)NC2CCN(C(c3c(C)cccn3)=O)CC2CO)CCC2CC1C2(C)C C1(CCC)(NC(=O)CCCn2c(C)csc2=O)CCCN(C(=O)C(F)(F)CO)C1 O=C1CN(C(c2ccc3c(c2)CCO3)=O)C2CCN(C(C3CC3F)=O)CC2N1 C1(CNC(C(C)SC)=O)CC2(CC2)CN1C(c1cnc(C(C)(C)C)nc1C)=O C1(C(=O)NCC2CC(F)(CNC(=O)C(C)CO)C2)(CSC)CC(F)(F)C1 c1(C(=O)NC2(COC)CCN(C(CC=CC=C)=O)C2)cc2n(c1)CCSC2 Cc1c(C(N2CCCCC2CNC(=O)CN(C2CCSC2)C)=O)cnn1C1CC1 c1(C(=O)NCCC(C)NC(=O)C(c2ccc(Cl)nc2)(C)C)ccc(N)c(F)c1F CC(C)(CC(=O)NC1CC(NC(c2coc3c(Br)cccc23)=O)C1)C(F)(F)F c1(C(=O)NCC(CN(C(c2cn(CC(CC)O)nn2)=O)C)O)cc(=O)n(C)o1 CC1CCC(NC(=O)CCC2CCCO2)CN1C(=O)CN1OC(C)(C)CC1=O C(=O)(CCC1=CCCCC1)OCCC(C)F C=CCCCCCCC(=O)NCC(CC(C)C)NC(C1(CCOC)CC1)=O c1(C(=O)NCC2(F)CC(NC(C3CC34CCOCC4)=O)C2)ncc(Cl)cc1F CC1NC(=O)CCC1Cn1cccn1.c12nnc(s1)NC2 CC(C)CC(F)(F)C(=O)NC1CC2(C1)CC2NC(=O)CN1CCCC(N(C)C)C1 CCCCS(=O)(=O)CC(=O)NC(C1CCCC1)CNC(=O)CC(C)N(C)C c1(CC)ccc(C(=O)N(C)CC2COCCN2C(c2occ(C)c2C)=O)nc1 N1(C(C)=O)CCC(NC(=O)CCc2cnnn2C)c2ccccc2C1 CC(C)S(=O)(=O)C(C)C(=O)NCC1(C(F)F)CCN(C(C2(C)CC2)=O)C1 c1(C(=O)NCC(CNC(CC2C(C)=NNC2=O)=O)(C)F)nc[nH]c2nccc1-2 c1(C(=O)Nc2scc(CN3CC(C(=O)OC)SCC3)n2)c[nH]c2ncc(Cl)cc12 N1(C(CC2CN(C(=O)OC(C)(C)C)C(C)(C)C2)=O)CCSc2ccncc21 C1(NC(CC)=O)CCN(C(C2(CNC(=O)CCOC3CCCC3)CCCO2)=O)C1 C1(NC(CCCCC)=O)CC12CCN(C(C1CCC(=O)N1CCC)=O)CC2 C1(C(N2CC3CN(C(CCCSC)=O)C3CC2)=O)Cn2c(C)nnc2CN1C C(CN=c1[nH]c2ccc(F)cc2s1)NC(c1ccnc(F)c1F)=O c1(C(N2CC3C(CNC(C=C4CCN(C)CC4)=O)(C3)C2)=O)cc2ccccn2c1 N1(C(Cc2c(C)ccs2)=O)CCC(C)C(CNC(c2cccc(CC#N)c2)=O)C1 C(=O)(C1=NNC(=O)C1)N1CC(CCNC(c2c(C)nc(CC(C)C)o2)=O)C(C)C1 c1(CC)noc(CCC(=O)NC(CN(C(=O)CC2COCCO2)C)CC)n1 CC(C)(O)C(F)C(=O)NC1CCCC1NC(=O)Cn1cc(F)ccc1=O Nc1cc(N2CCC(C(N3CCN(CC4COCCO4)CC3)=O)CC2)ncn1 CC1OC(C)C(C(N2CCOCC(NC(=O)CC3CCC(C)CC3)C2)=O)C1C N1(C(C2C(C)(C(C)C)C2)=O)CCC2(CC1)CN(CC1(C)CC1)CCO2 c1(NCC(CC)NC(=O)OC(C)(C)C)nccc(=NCC2(O)CCC2)[nH]1 c1(OC)nc(C)ccc1C(=O)NCC1CCCN1C(=O)CCc1ccc(C)nc1 c1(-c2c(C(=O)Nc3c(NCCC)cccc3)sc(Br)n2)ccc2c(c1)OCO2 Cc1cncc(C(=O)NC(C(=O)NCCCS(N)(=O)=O)c2ccco2)n1 c1(C(N2CC3C(CNC(c4ccc(COC)cc4)=O)C3C2)=O)ccc(N)cc1F N1(C(C2C(=C)CC2)=O)CCCN(C(C2CC(C(C)(C)C)=NO2)=O)CCC1 C1(C(N2CC(n3cc(-c4nccnc4C4CC4)nn3)C2)=O)(OC)CC(F)(F)C1 C=Cc1cnn(C)c1C(N1CC=CC(NC(=O)CCc2ccc(C)c(Cl)c2)C1)=O C1(c2cccnc2)(C(=O)NCC2C(NC(=O)CCOC3CCOC3)C2)CCCC1 C(=O)C(C)CCCOCCOC.C(=O)(C(C)(C)C)N.C1(=O)CCCN1CCC(C)C N1(C(C23CC(C)C2C3)=O)CC(O)CC1CNC(=O)CCc1ccc(F)nc1 C(CCN=C(NCCF)N1CCCC(O)CC1)=CC=C N1(C(CCCCC(C)=O)=O)CC(C2CCCN(C(=O)Cc3cnsc3)C2)C1 N1(CCn2c(C)ccn2)CCN(C(=O)C(C)COCC2CCCO2)CC1 N1(C(C(CCC#C)O)=O)CCC(C2CCN(C(c3ccc(Cl)o3)=O)CC2)CC1 N1(C(c2ccc(CC)o2)=O)CC2CCC1CN2C(c1ncoc1C(F)(F)F)=O C(c1ccc(F)cc1)=CC(N1CC=CC(NC(C(c2ccc(Cl)cc2)C)=O)C1)=O Cc1c(Br)ccc(-n2cc(C(N3CC(CO)(CC4CC4)C3)=O)nn2)c1C CC1=C(C)CC(C(N2CCCCC2CNC(c2cc(C3CCC3)[nH]n2)=O)=O)CC1 C1(C(=O)NCC(CNC(C(c2cccc(C)c2)O)=O)O)CCCC(C)(C)C1 Cc1coc(C(C)C)c1C(=O)N(C1CCCC1)CCCNC(c1coc(Br)n1)=O Cc1[nH]nc(Cl)c1C(=O)NCC1(F)CC(NC(=O)CC2(C)CCCO2)C1 C1(C(=O)OC)CCC(C2CCCO2)O1.c12ccccc1N1CCN(CC1)C2=O C1(OCCC)CCCN(Cc2cc(-c3cccnc3)no2)C1 C(CC(C(C)(C)C)NC(=O)Cn1ncc(O)nc1=O)N(C)C(C1CC1(C)C)=O CC(CC(=O)N1CCCC1C(O)CO)C(C)(C)NC(=O)COC(F)F c1(NC(C(c2cccc(C(C)C)c2)N(C2CC(=C)C2)C)=O)ccc2c(c1)OCO2 c1(C(=O)NC2CCCN(C(c3cncc(O)c3)=O)C2)c(Br)nc2n1CCC2 C1(NC(C(CC)N(C)C)=O)CN(C(C2(CO)CC2(F)F)=O)CC1CC C(C(CC(C)C)C(=O)NCC(C)NC(=O)CCCn1cccn1)OC C1(CNC(C2CC(C(=O)OC(C)(C)C)C2)=O)CC(O)CN1C(C1CC1(F)F)=O O(N(C(=O)C1C(O)CCN1C(C1CCN1C(C)(C)C)=O)C(C)C)CC C(N=c1nc(N2CCC(SC(F)(F)F)CC2)c2c([nH]1)COC2)C1(OC)CCOC1 Cc1ncsc1SCC(=O)NCC(C)(C)CC1CN(C(=O)C(C)CC2CC2)C1 C1(C(C(=O)N(CC(CO)C2CCC2)Cc2nn[nH]n2)F)CCCCC1 c1(C(=O)NC2C(NC(C3C(C)C3c3cccc(Cl)c3)=O)CCC2)ccc(=N)[nH]c1 C1(NC(c2n(CC)cc(Cl)c2)=O)COCCN(c2nccc(C#N)n2)C1 CC(C)C(C(=O)NCCCC(O)CO)C(C)NC(C1CC2CCCC2C1)=O N1(C(c2occ(C(N)=O)c2)=O)CCC(O)(CNC(=O)C(F)=CCCF)C1 CC1(C)COCCN(Cc2coc(C(F)(F)F)n2)C1 c1(OC)c(CN2C(C(=O)NCc3cc[nH]n3)CC(F)(F)C2)cccc1F C(=O)(C(F)CCC(C)C)NC1(CNC(c2cc(CC)c(Cl)cc2)=O)CC(OC)C1 N1(C(C)(C)C)CCN(C(c2n[nH]cc2NC(c2ccon2)=O)=O)CC1 C(=O)(C(C)(C)CCC#N)NC1(C(N2CCC(CC(C)C)C2)=O)CC(O)C1 c1(CC(=O)N(C)Cc2n(CCC)cnn2)ccc(OC2CCCC2)cc1Br c1(OC)cc(NC(C2CCCN2C(c2ccccc2C(F)(F)F)=O)=O)nc(Cl)c1 C1(N(C)C(C2(N(C3CC(CC(N)=O)C3)CCO)CCC2)=O)CCCNC1=O N1(c2ccnc(NC(c3ccn(C)n3)CC)n2)CCC(C2CC2(F)F)C1 C(CCC[Si](C)(C)C)OC(c1cc(C)ns1)=O c1(C(=O)Nc2ccc3ncsc3c2)cc(O)nc2cnccc12 c1(C(=O)NC(CC2CN(C(C3CC3[N+](=O)[O-])=O)C2)C)csc2cc(C(=O)OC)sc12 c1(C(=O)NCCN(C(C2CCCN(C(=O)OC)C2)=O)CC)nccc2n[nH]cc12 n1(CC(C(N2CCCN(C(c3c(C)snc3)=O)CC2)=O)C)ccc2ccccc12 c1(-n2ccc(C(=O)NC(CC=C)CO)n2)cc(C)ccc1C C(=O)(CCC(=O)NCC1(CNC2CCC(F)C2)CCC1)NCC C(c1ccc(O)cc1)=CCNC(=O)OC(C)(C)C.C(CCC(c1cccs1)N)NC=O C1(C(=O)NCC(C)NC(=O)C(O)CN2CCCC2)OCCOC12CCC2 C1(C(N)=O)CCC(OC(=O)Cn2cc(-c3ccncc3)nn2)C1 CCCCCC(=O)NC1CCOC(CNC(=O)CCc2cc(C)[nH]n2)C1 c1(CN(C(=O)NC2C(c3n(C)ccn3)C2)C2CC2)ccc(-n2cncn2)cn1 C1(C(=O)NCCC(C)OC)CCN(C(=O)CCc2cccnc2)C1C N1(C(CC)=O)CCN(C(=O)C(c2ccc(Cl)cc2)N(C)Cc2ccccc2)CC1 c1(C(=O)NCC2OCCCN(C(c3c(CC)c[nH]c3)=O)C2)c(C)ncn(C)c1=O c1(C(N2CCC(CNC(C(C(C)C)O)=O)C2(C)C)=O)ccc2cccc(O)c2c1 C1(C(=O)O)CN=C2N=C(CNC(C3CCC(c4n[nH]c(C5CC5)n4)O3)=O)NN2C1 CC1CN(C(C2COCCO2)=O)CC1CNC(=O)CNC1CC1 c1(C(=O)NC2(CC)CCCN(C(=O)C(C)O)C2)ccn2cc(C)nc2c1 N1(C(c2n(CC)nnc2)=O)CC2(NC(=O)C(C)CN(C)C)CCC1CC2 C1(C(=O)NC(C(c2c(C)cccc2)C)=O)CCN(C(=O)CCCC2CC2)C(C)C1 C(C)(C(N=c1cc(Br)n(C)[nH]1)c1nnnn1C1(OC)CC1)=C(C)C C1(CC(=O)NCC(C)CNC(=O)C(C)(Cl)Cl)CCCC1(F)F Cc1c(C(=O)NCC2C(C)CCN2C(=O)CCc2cccnc2)ccn1C(C)C c1(C(C)C)c(C(=O)NC2CC(O)(CNC(C3(C)CC3(Cl)Cl)=O)C2)cnn1CCO c1(C2C(NC(=O)Nc3cccc(C(C)(F)F)c3)C2)ccc(C#N)cc1 CC(C)(C(=O)NC1CCCC(NC(=O)COC2=CC(F)(Cl)C=N2)C1)C(F)(F)F CC(CC(=O)NCC#CC(=O)NCC1(C#N)CCC1)N(C)C c1(C(N(CCC)CCNC(c2ccnc(C(F)(F)F)c2)=O)=O)csc2nccn12 C(=O)(CCCCCCBr)N1CCCC(NS(CCOC)(=O)=O)C1 c1(CNC(N2C(C3(C(=O)OC)CCCCC3)CCCC2)=O)nccc(Cl)c1F C(=O)(C(O)(C(F)(F)F)C1CC1)NCC(CNC(C1(COC)CCC1)=O)C.C1CC1 N1(C(c2ccn(CC(C)C)n2)=O)CC(NC(C2CC3(CCC3)C2)=O)CC12CCC2 c1(C(N(C)CC2CCCN(C(c3cccc(C)c3)=O)C2)=O)cnc(Cl)c(C)c1 C(CCC(C)C)(C(=O)NCCC(O)CCC)NC(C(CC=CC)C)=O N1(C(C2(CC)CCC2)=O)Cc2ccccc2C(NC(=O)Cc2c(C)n[nH]c2C)C1 c1(COC)noc(CN(C)C(=O)NCCC23CC(C2)C3)n1 C1(NC(c2c(C)nc(NC(=O)CSC(F)F)s2)=O)CCS(=O)(=O)CC1 C1(CC#C)(C(=O)OCCSCc2csc(-c3ccc(C)cc3)n2)CCCCO1 N1(C(c2cncc(OC)c2)=O)CCN(C(=O)Cn2[nH]cnc2=N)CC1CF CCCC(C(=O)NCC(CC(C)C)NC(C1CC1C)=O)c1ccccc1 C(=O)(CC(C)CC(C)(C)C)N1CCC(CC)(NC(C2CCCCC(=O)N2)=O)CC1 Cn1ncc(NC(c2cc(Cl)c(Cl)s2)=O)c1-c1cn(CCC(F)(F)Cl)nn1 C(C(C)C(C)C(=O)N1CCCCC1Cc1ccc(F)cc1NNS(N)(=O)=O)OC N1(C(C(c2n(C)ccn2)(F)F)=O)CCC2(NC(c3cn4ccsc4n3)=O)CC2C1 N12CC3(CCN(CC3)C(=O)C=CCCCC1=O)C2.c1(CC)ccc(OC)cc1I c1(CCC(=O)NC2CCN(C(C3=C(C)CCC3)=O)C2C)nc2ccccc2s1 c1(C(=O)NC2(CC)CCCN(C(C3(O)COC3)=O)C2)cnc2ccc(C)cn12 N1(C(C2CC(OC)C2)=O)CCC2C(C1)CN2C(=O)COCC(=O)N(C)C Cc1cc(C2CCC2)ncc1C(N1CCCC1C(C)NC(=O)CC1CCOC1)=O C1(C(=O)NC2CN(C(CC)=O)C2)CC2CC1CN(C(c1coc(C)n1)=O)C2 C1(NC(C)=O)CCN(C(=O)CC(C)(C(=O)N(C)C)c2nn[nH]n2)CC12CCC2 CC1CNC(C)(C)CN1Cc1ccc(Br)c(Br)c1 C1(NC(c2cnc(CC)nc2)=O)CCN(C(=O)Cc2ccc(F)cc2C)CC1O CCCC(CCC)CCCC(=O)NC(C)C(CO)NC(c1cc(COC)on1)=O C1(NC(C2(NC(C3CCCCC3(F)F)=O)CSC2)=O)C2CCCCCC12 CCC(CC)C(C)C(=O)NC1CC(C)(NC(=O)Cc2cc(C)ccc2C(C)=O)C1 C1(CC(=O)NC(C)(CNC(=O)C=Cc2ccsc2)C2CC2)CCCC12CC2 C1(NC(c2c(CCC)nco2)=O)COC2CN(C(=O)C3=CCCCO3)CC12 C12(CNC(=O)Cc3ccccc3Cl)CCCN(C(c3ccnn3C3CC3)=O)C1C2 CN1CCOCC1C(N1CCC(C)(CNC(C2(CCS(N)(=O)=O)CCC2)=O)C1)=O CC1CC(CC(N2CCC(F)(F)C2)=O)CN1C(c1c[nH]c(=N)o1)=O CCC(C)C(O)CNC(c1coc(CNC(c2ccc(C#N)o2)=O)n1)=O Cn1ccc(C(=O)NCC2OCCC2C(N2CC(CC3CC3)C2)=O)n1 c1(CC)cccc(NC(=O)C(C)N(C(c2c[nH]c(=NC)o2)=O)C2CC2)c1F c1(OC)cc(OC)c(CN2CC3CC2C3C(=O)NCCN(C)C)c(OC)c1 N1(C(CNC(c2c(C)cccc2)=O)=O)CCC2C1CCN2C(C1(C(F)(F)F)CC1)=O CN1C(=O)NC2(CCCN(Cc3ccccc3CCCN(C3CC3)C3CC3)C2)C1=O c1(C(=O)NC2C(CNC(c3ccoc3)=O)CCC2)nnn2c1C(=O)NCC2 c1(C(N2CC(OC)C(NC(=O)C(F)C3CCC3)C2)=O)cc2cc(Cl)ccc2[nH]1 c1(C(N2CC(C(C(=O)OC)O)C2)=O)ccc(OCCCC(C)OC)cc1 C(=O)(C(F)CC(C)(C)NC(C12CC1COC2(C)C)=O)NC1(C(=O)OC)CC1 c1(OC)cc(C(N2CCCC(C(N3CC(C)C3)=O)CC2)=O)ccc1F c1(C(=O)NCCC(C)NC(=O)C(C)(C)CC2CC2)c[nH]c2cccc(F)c12 N1(C(C(=O)NC(C)CN(c2nocc2N)C)=O)CCC(C)OC(C)C1 c1(C(=O)NCC2OCCC(NC(C(C=C=C)C)=O)C2)ccc2c(O)ncnc2c1 CC1CCN(C(C2CC(C)CC(C)C2)=O)CC1CNC(=O)CCOCC(F)F N1(C(C(C=CC)O)=O)CC(NC(=O)CCSCc2ccccc2)C(C)(C)C1 C1(C(C)NC(=O)COc2ccsc2)CN(C(=O)COCP(C)(C)=O)CCO1 N1(C(C2CCCO2)=O)CCC2CCN(C(=O)CSc3cccc[n+]3[O-])C2C1 c1(OCC)cnnc(C(=O)NC(c2ccc(C)cc2)CNC(C2CCCS2)=O)c1 C(C(C(C)(C)C)NC(=O)Cc1cncnc1)NC(c1ccc(COC)s1)=O c1(C(C(=O)NC(C(C)NC(C2CC(CC)(CC)C2)=O)CO)O)cn(C)nc1C C1(O)(C(=O)OCC)CN(C(C2CCCN2C(=O)OC(C)(C)C)=O)CC1O C1(C)(C(=O)NCCN(CC(C)O)C(c2ccc(C(C)(F)F)cc2)=O)COCCO1 C1(CN(C(CC=CC)=O)CC)CCCN1C(=O)C(CC)SCC C(C)(CC(=O)NC(=O)CCCN1CCCC1)N(C(=O)COCC(C)C)CC N1(C(c2nccc(OC)c2C)C(=O)NCCC)CCC2(CC1)C(=O)NCCN2C Cc1ccc(C=CC(N2CC(NC(c3ccncc3F)=O)C(C(F)F)C2)=O)s1 N1(C(C=C)=O)CCc2cccc(COC)c2C1.c12cccc(c1)CCCC(=O)N2 c1(C(=O)NCC2(F)CN(C(CC)=O)C2)ccc(C)c(S(=O)(=O)CCO)c1 C1(C(=O)NCCCN(C(c2cc(COC)[nH]n2)=O)CC)CNC(=O)C(C)(C)C1 Cc1cc(C(N2CCN(C(=O)C(C)OC(C)(C)C)CC2CCO)=O)ccc1Cl C(=O)(CC1OCCc2sccc21)N(C1CC(C(=O)OC)C1)C1CC1 Cn1nnc2ccc(C(N3CCC4CC3CN4C(=O)Cc3ccco3)=O)nc12 C1(C(=O)NC(C2CCN(C(c3cccs3)=O)CC2)(C)C)(CC)CCNC1=O C12(C(=O)OCc3cc(OC)ncc3)CCN(C1)S(=O)(=O)C2 N1(C(CN(CC)CC)=O)CC2CC(NC(=O)C=CSc3ccccc3)C(C2)C1 c1(C(=O)NCC2CCNC2=O)noc2c1CN(C(c1ccc(Cl)c(Cl)n1)=O)C2 C1(C(N(CCCNC(C2(C(F)F)CC(=C)C2)=O)C)=O)CCCN(C)C1 c1(CNC(c2c(C)cns2)=O)ccc(C(C)NC(=O)CC2CC3C=CC2C3)cc1 Cc1cccc(C(=O)NCC(C2CCCC2)NC(=O)CC2CCC(=O)C2)c1C C(CC(C(C)C)NC(=O)COC1CCCOC1)N(C(C(CC)SC)=O)CC c1(C(=O)NC(CC)(C)CNC(c2nn(C)cc2C)=O)ccc(N)cc1S(N)(=O)=O c1(NCC(=CC(=O)NCCN(C(C2CCC(CC)O2)=O)CC)C)ccccc1F C123CCOCC1CN(C2)C(=O)CO3.O=C(C=CCl)NCCC(=O)N1CCCC1 c1(C(=O)NC(C2CCN(C(C(CC)OC)=O)CC2)C)cnc2cnn(C)c2c1 N1(C(c2c(C)c[nH]c2)=O)CCN(CC2CCN(C(=O)C(O)C3CCC3)CC2)CC1 C(=O)(CCCCCCS(N)(=O)=O)NCCC(C)NC(=O)C(C)(O)C1CCC1 c1(C(=O)NC(C)C(=O)NCCC#CCO)ccc([N+](=O)[O-])[nH]1 c1(C(CC(=O)NCCc2cccc(C#N)n2)O)nc2ccccc2[nH]1 C(=O)(C1Cc2ccc(Cl)cc21)NC1CC(C)(C)N(C(=O)CCc2cncnc2)C1 C1(CC(=O)N(CCC(C)NC(c2c(C(C)C)con2)=O)C)COCC1(C)C c1(CN2CC(C(=O)NCC3CCC3)SCC2)cc(Cl)c(Cl)nc1Cl C1(NC(CC=C)=O)CN(C(=O)C(C)=C2CCC2)C2(CCOC2)C1 Cc1nc(-c2ccc(CO)cn2)sc1NC(=O)N(c1cccc(Br)c1)C c1(C(=O)NC2CCN(C(CC(C)O)=O)CC2O)ccc2c(Cl)ccnc2c1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NCC(C2CC2)NC(=O)CN2CCCCCC2)c1 Cc1ccc(C(N2CC=CC2C(=O)Nc2csc(C3CC3)c2)=O)cc1C#N Cc1nc2c(C(=O)NC(CNC(c3cc(C)c(Cl)cc3F)=O)CO)cccc2o1 C1(CCCC)CN(C(=O)C(C(C)C)OCC)CCN1C(=O)CCc1scnc1C NS(=O)(=O)c1scnc1C(=O)NCCC1CN(C(=O)C(F)C2CCC2)CCO1 C(=O)(CC(C)C(F)F)N(CCN(C(CC1CC(C(=O)OC)C1)=O)C)C(C)C c1(C(=O)NCc2nc(C)[nH]n2)ncccc1NCc1cccnc1C(F)(F)F N1(CC2C(c3ccc(OC)cc3)C2)CC(C(N)=O)OC(C)C1 O=C1NCCCCC1N1CCN(C(C2CC=CC(n3ccnn3)C2)=O)CC1 c1(C(=O)NC2CC(F)(CNC(C3C(C=C)OCC3)=O)C2)c(C)sc2ccccc12 N1(C(C2C(CCC)CCC2)=O)CCCC2CN(C(=O)CC34CC(C3)C4)CC12 C1(NC(C(=O)NC(CC#C)CC(F)F)=O)CC2CCC(C1)N2C Cc1cccc(CC(=O)NCC(C)(O)CNC(=O)Cc2ccn(C(C)C)n2)c1Cl n1(CC(=O)NC(C2CCCCN2C(=O)CC2CCOC2)C)nnc2c1CCCC2 N1(C(c2nccc(OC)c2O)=O)CCC(CNC(=O)C2=NOCC2)C(F)(F)CC1 C=CC(C)(O)C(=O)N(C(CNC(c1cnc(OCC(F)(F)F)cn1)=O)C1CC1)C c1(C(N(C(C)CN(C)C(C2CC23CCC3)=O)C)=O)cn(C)nc1-c1ccoc1 c1(NC(C2C3C(=O)OCC23Br)=O)cc2c(cn1)COCC2 C(=O)(C(C)S(N)(=O)=O)NC1(CF)CCN(C(C2CC(C(=O)OC)C2)=O)C1 c1(SC)cc(C)ccc1C(=O)NC(CNC(=O)Cc1sc(O)nc1O)CO N1(C(C2OCCC(NC(c3c(C)nccc3)=O)C2)=O)CC2CCC(C1)N2C N1(CCC(=O)NC(CC)C(C)(C)O)C(=O)C2CC=CCC2C1=O c1(C(N2CCC(NC(C(F)=C(C)C)=O)C2)=O)cc(=O)c2cc(O)ccc2o1 c1(CNc2c(-c3ccc(OCCC)cc3)csc2)ccc(F)c2cccnc12 c1(CC)c(C(=O)NC2(C)CC(NC(=O)C3=COCCC3)C2)sc2ccccc12 c1(C(N2C(C(=O)N(C3C(CCOC)C3)CC)C(C)CC2)=O)ccc2cccnn12 C1(CNC(c2cnc(C(C)OC)s2)=O)COCCN(C(=O)CN2CSCC2=O)C1 Cc1sc(=O)n(CC(=O)N(CCCNC(C2C(C)(C)OC2(C)C)=O)C2CC2)c1C c1(C(C(=O)C(Cc2ccccc2)c2nc(C(N)=O)no2)(CC)O)cccc(C)c1 C1(C(=O)NCC2N(C)CCC2)COCCC12CN(C(c1ccsn1)=O)C2 C1(C(=O)NCCN2CC=CC2)(COC)CN(C(=O)Cc2nc(Cl)cs2)C1 C1(CC(=O)NCc2n(CCC)cnc2)N(C(=O)C(C)C2CCCC2)CCC1(C)C N1(C(c2nnc(SCC)s2)=O)CCN(C2CCCN(C(=O)C(C)OC)C2)C(=O)C1 CCCCC(O)C(C)C(=O)NCC1CCN(C(c2ccc(CSC)o2)=O)C(C)C1 N1(C(c2c(C)n(C)nn2)=O)CCC2(CCCCC2NC(=O)Cc2csc(Cl)n2)C1 N1(C(CCC2CC(OC)C2)=O)CCC(F)(CNC(c2nc(=N)cc[nH]2)=O)C1 C(CC(C)C(=O)NCc1cncc(C(=O)Nc2ccc(C(C)C)cc2)c1)=CC c1(N(CCCNn2ccnc2)C)nc2cc[nH]c2c(=NC2CC(CC)C2)[nH]1.CS S(=O)(=O)(c1cc(C)cnc1NCC(CO)OC)NCC(c1ccc(OC)cc1)O S(=O)(=O)(c1cnc2ccsc2c1)OC.c12ccc(cc1)OC(C)(OC)C2 c1(C(N2CC(C)C(NC(=O)C=C3CCC3)C2)=O)ccc(C#N)c(C(F)(F)F)c1 CC1CN(C(=O)C=Cc2cn[nH]c2)CC1(C)CNC(C1(CO)CCC1)=O C1(CNC(CCCOCC)=O)CC2CCC1N(C(c1ncc(F)cc1F)=O)C2 N1(C(c2cccc(CCC)c2)=O)CC2CC1CN2C(c1nnsc1C)=O c1(N(C)C)ncc(C(=O)NCC2CC(C)N(C(c3cnn(C(F)F)c3)=O)C2)cn1 N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CN(C(=O)C=Cc3cnc[nH]3)C2)C1 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CCC2CC(NC(=O)C(C)C)CCC2C1 O=C(N=c1ccn(CCN2CC(c3cn4ccccc4n3)C2)[nH]1)C12CC(F)C1C2 c1(C(N2CCCC(N(C(=O)C(C)C)CC)C2)=O)ncc(Br)cc1C N1(C(c2nccc(OC)c2)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1CO c1(C(=O)NCC(C)N(C(=O)C#CC2CC2)C)ccc2c(c1)OC(C)(C)OC2 CC1CN(C(=O)CC2CCC(=O)N2)CCCN1C(=O)CCCNC(N)=O N1(C(C(C=C)(F)F)=O)CC(CNC(=O)CCC2CCOC2)C2(CCC2)C1 Cc1cc(C)c(C(N2CC3(CNC(C4CCNC4=O)=O)CC2CO3)=O)c(C)c1 CS(=O)(=O)c1ccccc1CN1CC2C(Nc3ncnc4c(Br)c[nH]c34)C2C1 C(c1ccnc2ccccc12)=CC(=O)NC1CCCC(NC(c2ccns2)=O)C1 C1(NC(C(C)OC)=O)CCOC(C(=O)NC2CCC(C(C)C)CC2)C1 c1(NC(CCC(C)(C)NC(CCc2n(C)ncc2)=O)=O)cccc2c1CCC2 c1(C(N(C)CC2CCN(C(=O)COC(F)F)C2)=O)cccc(O)c1 C(=O)(CCC(=O)N1CCCCC1CNC(C1(O)CCSC1)=O)N(C(C)C)C C1(NC(C2(C)CN(C(=O)CC(=O)NC3CC3)C2)=O)CC2CC(O)C1C2 c1(C(=O)NCC2CC3CN(C(C(C)OCC)=O)CC32)cc2cnccc2[nH]1 C12(CNC(C(C(C)O)N(C)C)=O)CCC(C1)N(C(=O)CNS(N)(=O)=O)C2 C1(C(=O)NC2C(CNC(c3c(CC)csc3)=O)C2)CCC(=O)NC1 c1(Nc2cc(C)c(Cl)cc2Cl)cccc2ncccc12.C12C3C(CN1C2)C3 C#CC1CCCC(CNC(=O)CCCC(C)NC(=O)C(F)(F)C2CC2)C1 C(CCOCC)(C(=O)N(C(C)C(C)C)C)NC(c1cc(CC)on1)=O c1(C(N(C2CCN(C(C=C(C)C(C)(C)C)=O)C2)C)=O)cc(=N)[nH]cc1Br c1(OC(CC)C)ccc(O)cc1.c1ccc(C(=O)N(CCN(C)C)CCO)cn1 CCCC(C(=O)N1CCCC1(C)CO)NC(=O)CCc1cc(CC)no1 C(c1ccc2ncccc2c1)=CC(=O)NC(C1N(C(C=CC)=O)CCC1)C c1(C(C)NCC(N2CCSCC2)(C)C)ccc2c(c1)c(CO)cn2C N1(C(C2CN(C(C(C)=C(CC)C)=O)CC(C)C2)=O)CCC(F)(F)C(F)C1 C#Cc1ccc(C(=O)NC2CCC(C(=O)NCCC3CCOC3)C2)cc1C N1(C(C(C)C2CC2)=O)CCCC(NC(=O)COCCCF)CCC1 S(=O)(=O)(c1cc(C)cnc1N1CCN(C(=O)OC)CC1)N(C(CC)CC(C)O)C c1(C(N(CCNC(=O)C=Cc2ccsc2)CC)=O)c(F)cc(O)cc1F CC(C)C(C)C(C)CC(=O)N1CC2CC1C2NC(=O)Cn1ncc2cccnc12 Cn1nnc2c1CC(C(=O)N(CCNC(=O)C=Cc1nccs1)CC1CC1)CC2 C1(C)(CNC(C2(C(C)C)CCC2)=O)CN(C(C23CCC(C2)OC3C)=O)CCO1 n1(C(CC)C)ncc(C(=O)NCC(C(C)(C)C)NC(c2coc(Cl)n2)=O)c1C N1(C(C2CCCC(S(C)(=O)=O)C2)=O)CC=CCC2(CCOCC2)C1 C(=O)(CCC(=O)NCC(F)(F)Cn1cc(-c2cccc(F)n2)nn1)N(C(C)C)C c1(C(C)NC(=O)Nc2cccc(C3CC3)c2)ccc(Cl)c(F)c1 C1(C)(CNC(C=CC)=O)CCN(C(c2ccc(-c3ncc[nH]3)cc2)=O)C1 N1(C(CCCC)=O)CCC(O)(C(C)NC(c2cnc(-c3ccccc3)[nH]2)=O)C1 C1(C2CCN(C(=O)CS(N)(=O)=O)CC2)(NC(c2c(C)n(CCO)cc2)=O)CCC1 C(CC(=O)NCC(=O)NCC(CO)NC(=O)CC1CC1(C)C)NC(C)=O NCCCCCC(=O)NCC(C1CCC(F)(F)CC1)O CCCC(C)(O)C(=O)NC1CC1NC(c1ccc(N2CCCC2)nc1)=O C1(CC(=O)NC2CC(NC(C3CCC3OCC)=O)C2)(OCC)CCCC1 c1(CCC)nc(C)c(C(=O)NCCN(CCC)C(c2sc(C(C)C)nc2C)=O)o1 C(C(C(=O)NCCCCNC(=O)COC1CC1)NC(=O)CC)OCC N1(C(C(n2ccc(C)n2)(C)C)=O)CC2(CCC2NC(C2OCCN(C)C2=O)=O)C1 N1(C(CCOC(C)C)=O)CCC(OCCNC(=O)C(O)Cc2cnn(C)c2)CC1 C1(C(NNC(C)=O)=O)CCN(C(=O)OCC(C)(C)C)CC12CCC2 c1(OCC(N2CC(N(C(=O)CC34CCCC3C4)C)C2)=O)ccccc1CO.C1(C)CC1 CC(CC#N)C(=O)NCC1CCCN(C(=O)C(C)(F)F)C1 C(=O)(C1=NOC(C)C1)NCC(CC)NC(c1c(C)noc1C(F)(F)F)=O N1(C(c2cn(C)nc2O)=O)CCCC2(CCN(C(C3CC4CCC3C4)=O)CC2)C1 C12(NC(CC(C)(F)F)=O)CCCCCC1N(C(c1ccn3c1CCCC3)=O)CC2 C(=O)(C1(C)CCn2ccnc21)N1CC(C(C)NC(c2oc(CC)c(C)c2)=O)C1 C1(C(N2C(C)CCC2)=O)CN(C(c2cn(C)ccc2=O)=O)CCN1C c1(C(N2C3C(NC(C4CC5CC5C4)=O)C(CC3)C2)=O)cccc2nn[nH]c12 S(=O)(=O)(c1c[nH]c(C(N2CC(NC(C3CC(C)(C)C3)=O)CC(C)C2)=O)c1)NCC c1(OCC(C)C)cccc(F)c1NC(N1CCNCC1C(C)C)=O N1(C(c2ncc(C)cn2)=O)CC2CCC1C(NC(C=CC(=O)OCC)=O)C2 N1(C(C2C(OCC)CC2)=O)CCC(C2CC2)C1C(=O)NCc1cccn(C)c1=O N1(C(C(CCC#C)NC(c2cnsc2C)=O)=O)CCCC(C)(C)C1C n1(CCSC)nnnc1C(c1occc1C)NCCc1cc(C)no1 CC(C)CC(CNC(C1CCC2(CCC2)C1)=O)C(=O)NC1CC(C)CCC1O c1(C(N2C(CCNC(c3nc(CCC)oc3)=O)CCC2)=O)cc2c(s1)CCC2 CON(CCC(=O)N1CCCC1CC(C)C)C(=O)C1CN2CCN1CC2 c1(CNCCc2ccc(-c3c(O)cc(O)cc3O)cc2)ccc(F)c([N+](=O)[O-])c1 N1(C(=O)C(O)C(F)(F)F)CCN(C(=O)C(F)(F)c2ccncc2)CC(O)C1 N1(C(CCSCCCC)=O)CC2CC2(CNC(=O)CN2CCC(C)CC2)C1 C#Cc1cncc(NC(=O)C(O)(C(C)NC2CN(C3CC3)C2)c2ccccc2)c1 c1(SC)ccc(C=CC(=O)NCC2CC(NC(=O)CCNC(C3CC3C)=O)C2)s1 C1(NC(CCn2c(C(C)C)ncc2)=O)(CNC(=O)C=CCF)CCCCC1C c1(CC(=O)NCC(=O)NC(CC=C)CNC(=O)C=CC(F)(F)F)cccc(C)c1 c1(CC(=O)NCC2CCCCN2C(=O)C(F)=C2CCC2)ccc(C(F)F)cc1 N1(C(c2scc(S(N)(=O)=O)c2)=O)CCC2CC(C1)CN(C(=O)CCCF)C2 C1(CNC(N(C(CC)C)C)=O)N(C(=O)OC(C)(C)C)CC12CCOCC2 c1(CN2CCCC(C)(CNC(c3ccc(SC)s3)=O)C2)ncccc1S(C)(=O)=O c1(C(=O)NC(CC(C)C)CNC(=O)CCCN(C)C)ccc2c(c1)C(=O)NCC2 N1(C(c2cccc(OC)c2)=O)CC2CCCC(C1)N2C(C1CCC(C)C1)=O N1(C(C2CC(=C)C2)=O)CC2CCC1CN(C(c1nccc(OC)c1OC)=O)C2 N1(C(CNC(C=C)=O)=O)CCOC(c2cn(C3CCOCC3)nn2)CC1 Cc1cc(C#N)cc(C(C2CCC(C)(C)CC2)O)c1N.C1CC(=O)N1CCO c1(OC)ccc(CN2CCNCC2)c(NC(=O)CC23CCC(C2)NC3)c1 c1(OC)cc(N)c(C(N2CC(NC(=O)C3=NOC(C)C3)CC(F)C2)=O)cc1OC N1(C(c2cnc(OC)nc2)=O)CCCN(C(=O)COc2cccc(C)c2)C(C)C1 C1(CNC(C(C)SC)=O)Cc2ccccc2CN1C(=O)C(=O)NCCNC(C)=O c1(C(C(=O)NCCCN)NC(=O)OCC)ccc(F)cc1 CC1C(C(=O)NCC(C)(C)CC(N2CCC3(CC2)CSC3)=O)=NOC1C c1(C(=O)NCC(CNC(C(C(C)C)O)=O)(C)O)cc(C(F)(F)F)cc(N)c1 c1(CN(C(C(=O)N(C(CC)CO)CCc2ccccn2)=O)C)cc(Cl)ccc1Cl N1(C(c2c(C)nc(C)[nH]2)=O)CC2CN(C(c3ccn4nccc4n3)=O)CC2(C)C1 C1(N(C(COCCCOC)=O)C)CCCN(C(c2n[nH]c(C)c2Cl)=O)C1 c1(C(N2C3C(NC(CSC(C)(C)C)=O)CC(C3)C2)=O)cccc(C#CCO)c1 N1(C(C(=O)N(C)C)=O)CCCC(C2CC2NC(c2ccccc2C(F)F)=O)C1 N1(C(C)=O)CC(C)(C)CC1NC(=O)NC(C(=O)NC)C(C)C1CCOC1.C(C)(C)(C)O Cc1nc2ccc(C(=O)NCC3COC(CN=c4cc(F)nc[nH]4)C3)cn2c1N C1(CNC(C2CCOC(C3CC3)C2)=O)COCCN1C(c1ccc(O)cc1)=O N1(C(=O)Cc2ccoc2)CCC2(CC1)CN(C(=O)CC1CC=CCC1)CC2CO N1(C(c2n(CC)ncc2Br)=O)CC2CC(C1)N(C(=O)C=CC(C)(C)SC)C2 O=C1N(C2CN(C(=O)C(F)CC3CCOC3)C2)C(=O)N1.C1(N)CCCC1 N1(C(c2cn(C)nn2)=O)CC2(C1)CN(C(=O)C(CO)C(C)(C)C)CCO2 CCC(C)(CC)C(=O)N1CCC(C)C(CC(=O)NCC2CCCCC2)C1 CC1(C)CC(C(=O)NC2CC3CCC2C3)CN1C(=O)CCc1ccc[nH]1 c1(C(=O)NC2C(NC(c3nc(C(C)OCC)sc3)=O)C2)ccc(C)nn1 C1(CCC)(NC(=O)CS(=O)CC)CCCN(C(c2c(C(F)(F)F)noc2C)=O)C1 C1(NC(C(C)CC2CC2)=O)CC(F)(F)CC1NC(c1cnoc1C1CCC1)=O C(CC(CNC(C1CC1OC(C)=O)=O)NC(=O)CCC1CCC(=O)N1)OC N1(C(C2CNC(=O)N2)=O)CC2(C1)CN(C(C1CCc3ccnn3C1)=O)CCO2 c1(COCCOC)ccc(NC(N2CCN(Cc3ccccc3)CC2)=O)cc1F N1(C(CC(CNC(C(CC)CC)=O)(C)C)=O)CC2CCC(CO)C2C1 C(c1ccccn1)=C(C)C(=O)NC1CC1NC(c1cccc(SCC#N)c1)=O Cn1nc(CC2(C)CCCN2)c(Br)c1Cl.C1(N2CCCC2)CCCN(C=O)C1=O N1(C(c2c(OCC)cccn2)=O)CC(CO)C2(CCN(C(=O)CSSC)CC2)C1 C1(CNC(c2cc(CNC(=O)CC3CSCCO3)oc2)=O)CC2(CCCO2)C1 CC1CN(C(=O)CC2(C)OCCO2)CC1CNC(c1cnc(C(C)(C)CF)o1)=O c1(CNC2CC(C(=O)NCCc3cscn3)C2)ccnc2ccccc12 Cc1cc2ncc(CNC(N3CCC(CN(C)C)C3)=O)cn2n1 C1(CNC(c2cc(C)c(C)[nH]2)=O)CCC(F)(CNC(=O)CC2CNC(=O)C2)CC1 C1(NC(=O)CCC(F)(F)F)CN(C(C2(O)CCN3CCC2C3)=O)CC12CCC2 c1(CC(=O)NCC2C(CNC(=O)OC(C)(C)C)C2(F)F)ccc(F)c(F)c1 N1(C(c2cnc(O)o2)=O)CCCCC1C1CCN(C(c2ncccn2)=O)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCC1(CN(C(=O)CC2COCCO2)C)CC1 Cc1nc(C2CC2)sc1C(=O)NCCN(C(=O)CC1NC(=O)NC1=O)C1CC1 N1(C(c2n(CC)ccc2)=O)CC2C(NC(C3CCN(C)C3=O)=O)C2C1 C(=O)(C(C(C)C)n1cccc1)NC(CNC(Cc1cnc(C)s1)=O)C C(CCC(N)=O)(C(=O)N1CC2CC1C2NC(C1CCS(=O)(=O)C1)=O)N(C)C CCCCCC(O)C(=O)N(CCC(N1CCC(CC2CC2)CC1)=O)CC1CC1 c1(-c2cn(C(C)C(=O)N(C3CC3C)C3CC3)nn2)cc(Cl)c(Cl)cc1Cl C1(C(=O)Nc2c(C)ccc(F)c2)CC2CCCCC2N1C(C1CCCS1)=O Cn1cc(NCC2CN(C(=O)CC(O)C3CCCC3)C2)c(O)nc1=O NS(=O)(=O)C1CCN(c2cc(N3CC4CC3CS4)ncn2)C1 C(CCCCCNC(C1(n2cnnn2)CC1)=O)NC(CC=C)=O CCCC(CC)(c1ccccc1)NC(=O)CCSCc1ccccc1 N1(C(c2cc(C)n(CC(=O)OC)c2C)=O)CC(C2CN(C(=O)C3=CCOCC3)C2)C1 CN1CCCC(C(N2CC3C(CNC(c4cocc4C(N)=O)=O)C3C2)=O)C1 N1(C(C2N(C(C3C(C(N)=O)C3)=O)CC(=O)NC2)=O)CCCCC2(CCC2)C1 N1(C(c2n(CCCC)ncc2)=O)CC(NC(=O)Cc2cnnn2C)CCC1C N1(C(C)=O)CCC(C(C)NC(=O)CC2(C(C)OC)CC2)CC1.C1(=O)CN1 N1(CC(N2CCC(CNC(C(C)Cn3cccn3)=O)C2)=O)CCCNC1=O Cc1ccc(NC(=O)C2=CCC(NC(c3sccc3CO)=O)C2)c(C)n1 CC1CCC(C)(Nc2ccc(C3CCN(C(=O)OC(C)(C)C)CC3)cn2)C1 N1(C(C(C(CC)C)OC)=O)CC2CC(NC(=O)CNC(C)=O)CC2C1.C1(C)(O)CCC1 c1(C(=O)Nc2n(C)nc(-c3ccccc3)c2)cccc([N+](=O)[O-])c1O O(NC(=O)C(n1cccn1)NC(=O)C(C(C)C)C1CCC1)C(CC)CC CC1(NC(c2[nH]ccc2C2CC2)=O)CCCCC1C(=O)NCc1ncon1 N1(C(CNS(NC)(=O)=O)=O)CC(NC(=O)C=Cc2cccs2)C(C)C1 c1(NCC(N2CCC(NC(COCCCC)=O)C(C)C2)=O)cc(C)c(Cl)c(C)c1 N1(C(CSc2cn(C)nc2)=O)CC2CCC1C1CN(C(=O)Cn3ccnn3)CC21 c1(C(=O)OCC(C2(C#C)CC2)=O)ccc2c(c1)C(=O)NCC(C)(C)O2 C12CC3(C1)CC3NC(=O)CC1(CCC1)O2.C1(NC(C=CC)=O)CCC(C(F)(F)F)O1 Cc1cc(C(N2CC(NC(c3nnn(C)c3C)=O)C(C)(C)C2)=O)c(N)cc1F C1(C(=O)N)OCC2CN(c3ccncn3)CCC12.O=C1OCC2(CCN(C(=O)CF)CC2)C1 c1(C(N2CC(CNC(C3CCCC4(CC4)C3)=O)C(O)C2)=O)cc2ncccn2n1 c1(C2CC(C(=O)NC(=O)C3=CCCC3)(NCNC(=O)OC(C)(C)C)C2)ccc(Cl)cc1 C(=O)(C(CC)CC(C)C)N1CCCC(C)(C(N2CC(CC(C#C)C)C2)=O)C1 N1(C(CC2CCC(C)C2)=O)CCC2(CCC(NC(C3(C)CCSCC3)=O)C2)C1 c1(C2(C)CC2)cc(C(=O)NC(CNC(=O)Cn2cc(CO)nn2)CO)no1 N1(C(C(F)=CCC)=O)CCC(CC(C)NC(=O)CCCNC(C)=O)CC1 CCCCC(C(=O)N1CCCC1CCNC(=O)C(C)N(C)C(C)=O)NC(N)=O Cc1ccc2c(N3CCOC(C(N)=O)C3)nc(N3CCOC4(CCC4)C3)nc2c1 c1(C(N2CC(CNC(CC(CC)C)=O)CC2(C)C)=O)ccc2c(C)noc2c1 CCCC(C)(CC)C(=O)NCCNC(C1CCN(Cc2nnn(C)c2N)CC1)=O C1(C(=O)NCCN2CCC(NC(c3scnc3C)=O)CC2)(OC)CC2CCC1C2 C[Si](C)(C)C1(NC(C2CCC(C3CC3)N2C(=O)CCCNC(N)=O)=O)CC1 c1(C(N2C(C(N3CC(C)(C)C(O)C3)=O)CC3(CC3)C2)=O)ccc2cccnn12 Cc1cccc(C2(C(=O)NCCC3CN(C(c4cscc4C)=O)C3)CCCC2)c1 C(=O)(C1=CC2(CN(C(=O)CC3C(=O)NN=C3C)C2)OC1)N(CC(F)F)CCOC C1(C(=O)Nc2ccc(OC)c(F)c2)CN(C(=O)C2=CCOCC2)C2(CCC2)C1 c1(C(N(C(C)CCNC(C2CCCOC2C)=O)C)=O)cccc(S(C)=O)c1 C1(NC(c2ncc(C)[nH]2)=O)CN(C(=O)CC2(N(C)C)CC2)C2CCCC12 C1(NC(=O)CCCn2cc(CC3C4CCCCCC34)nn2)CC(O)C12CCC2 S(=O)(=O)(c1ccc(Cl)s1)NC(C(N1CC(NC(CN(C)CC)=O)C(C)C1)=O)C c1(C(N2C(CC(CN(C)Cc3c(C)nc[nH]3)C)CCC2)=O)c(C)cccc1C C(N=c1[nH]c2c(c(=NC3CC4(CCCC4)C3)[nH]1)CCCCC2)c1n(CCC)ccn1 N#Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CC(C(F)F)C1 C(c1ccc(F)c(Cl)c1)=CC(=O)NCC(CN(C)C(c1cn2c(n1)CCC2)=O)O C(c1cc(F)c(F)c(F)c1)=CC(=O)N(CCN(C(C1OCC1(C)C)=O)CC)CC C#CCCCCCC(C(=O)NC(C)CC)N1CCN(c2ncccc2C)CC1 C(=O)(C1CCCc2sccc21)N1CC2CC(CNC(C(C)(C)C)=O)C2C1 C(=O)(C(F)CCC(C)(C)C)NC(C(C(=O)N1CCC(OC)C1C)C(C)C)C CCC1C(=O)N2CCCC2CN1C.c1(S)sccc1C C1(CNC(c2cnc(CC)nc2)=O)CCC2CN(C(=O)C(C#N)CC)CC12 c1(C(N2CC=CCC2(C)C)C(=O)NCCCSC)ccc(F)c(C)c1 C=CCCCC(C(=O)NCC=CC1CC1)NC(c1cc(C#N)n(C)n1)=O N1(C(C2CN(C)C(=O)C2)=O)CC(C(=O)NC2CC2CC(N)=O)CC1(C)C c1(C=O)nccnc1C.C12(C(NOCCC=C)=O)CC(N(S(C)(=O)=O)CC=C)(C1)C2 n1(CC)ncc2c(NC(CNC(C3CC34CCOC(C)C4)=O)C(C)C)ncnc12 C1(C(C)NC(=O)CC2(C)CC2)CN(C(c2ccc(C(F)(F)F)cc2)=O)CCO1 N1(C(=O)NCC(CC2CCCO2)OC)CCN2C(CNS2(=O)=O)C1 C(=O)(C(C)C(C)O)NCCN(CCOC)C(c1sccc1C(F)F)=O c1(C(=O)NC(CNC(C(C)OCCOCC)=O)C)c(OC)n[nH]c1CC C(=O)(CC(=O)NC(Cc1cn[nH]c1)C(=O)NCC(CC)n1cccn1)NCC#C c1(NC(c2oc(C)c(Br)c2)=O)cnc(F)cc1C(=O)NC1CC1 C1(C(N2CC(NC(c3cc(C(=O)OC)cn3C)=O)C2)=O)CCOC2(CCCC2)C1 c1(C(CNC(c2c(CC)c[nH]c2)=O)NC(C2CCCS2)=O)c(F)cccc1F C1(CNC(C(c2cn(C)nc2)NC(c2cc(CCO)on2)=O)=O)CCCCCC1 c1(C(=O)NC(C2CCCCN2C(=O)C2=CCCS2)C)cc(C#N)ccc1Cl N1(C(c2cncc(SCC)n2)=O)CC2CC3CC2C1C3NC(=O)C1=CCSC1 N1(Cc2ccn(CC)n2)CCCC(C(N2CCC(C(=O)O)C2)=O)C1 C12CN(CCO1)C(=O)NC2.C1(C)(C(=O)OCC)COC(c2ccccc2)O1 CC(CO)(CO)C(=O)OCC(c1ccnn1CC(F)(F)F)=O c1(C(N2C(CCCC)CCC2)C(=O)NC(C)(C)C)nccc(OC)c1C c1(CC)oc(C(N2CCCC2C(C)(C)NC(C2C3CCN2CC3)=O)=O)cc1C C(=O)(CCCC(C)=O)NCCCCN(C(C=CC=CCC)=O)C C1(CN(C(=O)C(c2ccncc2Cl)NC(=O)OC(C)(C)C)CC)CCS(=O)(=O)C1 C=CC(C)(CC)C(=O)N1CCC1Cn1cc(C2(C)CCCN2C)nn1 N1(C(c2cnc(CNC(C(CC(C)C)O)=O)nc2)=O)CCC2(CC1)CSC2 c1(C(=O)NC2C(NC(c3cc(CC)nn3C)=O)CCOC2)cccc2nsnc12 c1(OC)cc(N)ccc1C(=O)NCC1CCC(NC(c2cc(O)nn2C)=O)C1 Cc1nc(N)c(CCNC(=O)NCCC2(C)COCCO2)c(O)n1 N1(C(C23CC(C)C2C3)=O)CC(CNC(=O)CC2CS(=O)(=O)C2)OC(C)(C)C1 CCC(CC)C(C)C(=O)NCC1CN(C(c2ccc(C(C)(C)C)cc2)=O)CC1O C=CC(CCC)CC(=O)NCC(O)CCNC(c1cc(CO)n(C)n1)=O C#CCC(C(=O)N1CC(O)(CNC(C2CCOC2c2cccnc2)=O)C1)C1CC1 C(C(C)(CO)NC(c1ccn(C(F)F)n1)=O)NC(CNC(C)=O)=O C(N=c1[nH]c(=NCCc2ncccc2F)[nH]c2c1CSC2)c1n(CC)c(C)nc1 c1(NC2CN(C(C)C)C(CO)C2)ncc(S(=O)(=O)NCC2CCCC2O)cc1Cl C(=O)(C1=NOC(C)(C)C1)NCC1C(NC(CNc2ccc(OC)cc2)=O)COC1 c1(C(=O)NCC(C)CNC(=O)CNC(N)=O)cccc2[nH]ccc12 Cc1oc(CNC(C2(CN(C)C)CCC2)=O)nc1C(=O)NC(C)Cc1nc[nH]n1 C1(CNC(CSCCCC)=O)COC(CNC(=O)Cc2n[nH]c(C)n2)C1 c1(C(=O)NC(C)C(C)NC(c2cc(N)cc(O)n2)=O)cccc2c1CC(=O)N2 N1(C(CCCC=C)=O)CCC2CN(C(=O)CCS(C)(=O)=O)CCC12 c1(C(N(C2CN(C(C3(C)CCN(C)CC3)=O)C2)C)=O)cc(Cl)cc2c1NCCC2 C(CCCC(=O)NCCOC1CN(C(c2cccc(CN(C)C)c2)=O)C1)=CC CCCC(C)CC(=O)N1CC2CC1CN2c1ncc(C)c(O)n1 N1(C(c2nnc(N(CCCC)C)n2CCOC)C2CC2)CCC2(CCCNC2)C1 c1(CNC(=O)NC(c2ccc(Cl)s2)C)cccc(S(C)(=O)=O)c1 C1(C2(C(=O)OC(C)(C)C)CC(C)C2)CN(C(=O)NCCCNC(N)=O)CC12CCC2 C1(CC)(NC(C2CCC(F)C2)=O)CCN(C(=O)CC2=CCCC2)CC1 N1(C(CCCOCCOC)C)CCC(C)(CNS(C)(=O)=O)C1 CC1CN(C(C2(N(C)C)CC2)=O)CC1NC(C1CN(C)CCO1)=O C=C(C)C1OCCC1C(=O)NCC(=O)NCC(=O)NC1CCCN(C)C1=O n1(CC(=O)NCCCN(C)C(c2ccc(C(F)(F)F)cn2)=O)cc(C#N)cn1 C(=O)(C(C)(C)S(C)(=O)=O)N(CCNC(C1CC(C(C)C)OCC1)=O)C(C)C N1(C(c2c(OC)cncc2)=O)CCC2CN(C(=O)C(C)CC(C)C)C2C1 N1(OCCCSc2ccccc2)CC(C(=O)NCc2nc(C)sc2)CC(F)(F)C1 CC(C(=O)NC1CCC1NC(c1csc(C(F)F)c1)=O)C(C)(C)C c1(C(=O)NC2CCC(CNC(c3ccsn3)=O)CC2)ccnc2ncccc12 N1(C(c2scc(C)c2Cl)=O)CCCCC2(CCN(C(=O)C=C(Cl)Cl)C2)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(O)(C2(CNC(=O)C3=CCCCC3C)CC2)C1 c1(C(=O)NCC2C(C)(C)CN(C(C3(CO)CCCO3)=O)C2)cc2c([nH]1)CCCC2 C=CC(CCC)CC(=O)NC1(CO)CC(C(F)F)C1.C(=O)(CC(=O)OC)NC N1(C(c2csc(C(C)(C)C)c2)C(=O)N(C(CC)C)C2CC2)CCC(C)(F)C1 N1(C(C2C(n3cc(CS(C)(=O)=O)nn3)CCC2)=O)CC2C(Br)C2C1 CC1CCN(C(=O)CCCC(C)(C)C)CCN1C(c1ccc(N(C)C)cc1)=O c1(C(=O)NC2C(CNC(=O)C=C3CCCCC3)COC2)ccc(CO)c(F)c1 O=S1(=O)CCN(C(=NCCF)NCC(F)(F)C2CCC2)CC1 CC1(C)C(=O)CC1C(=O)NCC1CCCCN1C(C1C=CCCC1)=O c1(C(N(C)CC2COCCN2C(=O)C(O)C2CC2)=O)c(F)cc(F)cc1Cl N1(C(Cc2c(C)scc2)=O)CCC(C)(NC(=O)CSCCC#N)C1 C1(Nc2cc(N(CC(C3CC3)OC)C)ncn2)CCC(N=[N+]=[N-])CC1 c1(CNC(C2C(OC)CC2)=O)ccnc(N2CCN(C(=O)CCC3CC3)CC2)c1 c1(CC(=O)OC)cccc(C(=O)N(C2CC(NC(c3c[nH]nc3C)=O)C2)C)c1 c1(CC(=O)NCC=CC(=O)NC2COCC2CN2CCC2)cccnc1Cl C(=O)(C(F)(F)C(C)O)NCC12C(CN(C(c3c(C)nsc3N)=O)C1)C2 C1(CC=C)(C(=O)NC(CNC(C2CCCCN2CCC)=O)CC=C)CCOCC1 N1(C(c2cnn(C(F)F)c2)=O)CCCN(C(c2cnc(S)[nH]2)=O)CCC1 N1(C(c2cc3sc(Cl)cc3s2)=O)CCC2CN(C(=O)Cc3ccon3)CC2C1 C1(CN(C(COCCC)=O)C)CC(F)CN1C(C1CC2(CC2)CO1)=O N1CCCCC1C1(C(F)(F)F)N=N1.C1(CC=O)(C(C)C)CCC1 N1(C(c2ccc(OC)nc2C)C(=O)NC2CC(CC)C2)CCC2(CCOC2)CC1 c1(C(=O)OCC)cnc(C)[nH]c1=NC(C)CNC(=O)Cn1nnc(C)n1 c1(C(N2CCCC(CNC(c3n[nH]c(C)c3Cl)=O)C2)=O)ccc2[nH]c(=N)sc2c1 N1(C(C2=CC(C)(CC)C2)=O)CC2(CCC(NC(c3cc(C)ns3)=O)CC2)C1 n1(CC)nc(C)c(C(=O)NCC2COC(CN)C2)c1C(F)(F)F c1(C(=O)NC)cccc(C(N2CCCC(N(C(=O)C(C)NC(N)=O)CC)C2)=O)c1 C(CC(=O)NCC1(CO)CC1(C)C)(C(F)F)OC N1(C(C2C(CC)C2)=O)CCC2(CCCC2CNC(C2CCCC(CF)C2)=O)CC1 C1(NC(C(C2CN(C(=O)OC(C)(C)C)C2)O)=O)CCCCC1 c1(C(=O)NC2CCC(NC(C3CC34CCOCC4)=O)CC2)cc2c([nH]1)CCOC2 c1(C(=O)NC2C3CCN(C(CC4(O)CCN(C)CC4)=O)C32)ccc(S(N)(=O)=O)o1 c1(C(=O)NC2C(NC(c3cnn(CC)c3C)=O)CCC2)c(F)ccc(O)c1F C1(NC(=O)C=CC(=O)NC2CC2)CN(C(=O)CC2C=CCCC2)C2CCCC12 C(=O)(C(C)(C)CC(C)C)N1CC(NC(C2(C(=O)NC)CC2)=O)C(C(F)(F)F)C1 C(=O)(CCS(N)(=O)=O)NCc1c(C(N2C3(C(=O)OC)CC3CC2)=O)occ1 c1(CC)c(C(=O)NC2CN(C(c3sc(C(C)C)nc3C)=O)CC2C)nnn1CC C1(CCOC)CN(C(=O)CC2COC(C)(C)C2)CCN1C(=O)CSCCC(C)C CCC(CC)(CC)C(=O)N1CCC(NC(C2CC(=O)N(O)C2)=O)C1 c1(CNC(CC2(C#C)CC2)=O)ocnc1C(=O)NCCC(O)COCC C#CCC(CC(=O)N1CCC1C=C)NC(=O)C(C)(O)C=C C=CCC(CC)C(=O)N(CCC(C)NC(=O)C=C1CN2CCC1CC2)C n1(CC)cnc2c(NCC(C)(C)C3CCCO3)nc(N3CC4CC3CC4=C)nc12 C1(O)(CCNC(CCCOCC)=O)CCN(C(C2CCS2(=O)=O)=O)CC1 C(c1ccc([N+](=O)[O-])s1)=C(C(N1CCN(C(C=NOC)=O)C(C)C1)=O)NC(C)=O c1(C(=O)NCCN(C(=O)CNC(C2(F)CC2)=O)CC)ccoc1 C1(NC(Cc2c(C)occ2)=O)CC=C(C(=O)NCc2cnccn2)C1 C1(C(N2C(C(=O)NC)CCC2)=O)COCCN(C(=O)CC2CC(C3CC3)C2)C1 n1(CCCC(CCCC)O)cnc2c(N3CCCCCC3)ncnc12 C1(CC(N2CCC(C(C)NC(c3nn(CC)nc3C)=O)C2)=O)CCCCC1(F)F C(=O)(C1=COCCO1)N(C(CN(C(c1ccc(C(C)=O)nc1O)=O)C)C)C CN=c1nc(N(C)Cc2cccc(F)c2F)[nH]c(=NCCC(=O)N(C)C)[nH]1 C(=O)(C(C)(C)C(C)(F)F)N1CCOCC(CNC(CC(C)(C)N(C)C)=O)C1 c1(C(C)(C)C)nc(CCCCC(C)(C)c2ccccc2)n[nH]1.C(=O)(C(=O)N)CCN CN1CCOC(C(=O)N(CCCNC(C2CC3CC3C2)=O)Cc2cccnc2)C1=O Cc1ccc(C(C)NC(c2conc2C(C)NC(=O)C#CC(=O)N(C)C)=O)nc1 Cc1cc(C(=O)NC2CN(C(=O)CCCn3ccnc3C)CC2F)oc1C C12(CNC(=O)C=CCO)CCC1CCN2C(c1ccc(-c2cccs2)o1)=O C1(F)(CNC(c2c(C)nc(-c3nc[nH]n3)s2)=O)CCCN(C(=O)C(Cl)=CCl)C1 CCCCS(=O)(=O)CC(=O)NCC1C(C)CCCN1C(=O)C(C)O c1(CN2CCN(C)C(CC3CC3c3ccccc3)C2)n[nH]c2ccc(F)cc12 C(=O)(CCCCCN(C)C(C1(C)CC1(C)C)=O)NCc1nnc(CC)o1 Cc1ccc2sc(N3CCC(Oc4ccc(OCCCO)cc4)CC3)nc2c1 N1(C(C(C)OCC=C)=O)CC2(CCCN(C(c3ncncc3N)=O)C2)C1 C1(NC(c2cnn(-c3ccccc3)n2)=O)CCCCN(C(=O)CC2CCC2)CC1 c1(C(=O)NCC2CCCCN(C(CCOCCC)=O)C2)cnc2c(c1)CCCC2 CC1CC(NC(c2cc3n(c2)CCC3)=O)CCN1C(=O)C=Cc1ccncn1 c1(C(=O)NCC2(OC)CN(C(=O)C(F)CC3CCOC3)C2)ccc(N)cc1Cl Cc1cnc(C(=O)NCC2CC2C(=O)NC(CO)C(C)C)c(C)c1 C1(NC(CC=C)=O)CC(C)CN(C(=O)C=Cc2ccc(C)o2)C1 CC1CCCN(C(c2ccc(C3CC3)o2)=O)C1CNC(C1CC(C)(O)C1)=O CC1=C(C(=O)NC2CCCC(CNC(=O)CC3CN(C)C3)C2)CC1 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(CC(C)NC(C2=C(C)OCC2)=O)C1 C1(NC(=O)CC2CC2)CN(C(c2cc(-c3cccs3)on2)=O)CC12CC2 CCCCCCCCC(=O)N(CCNC(C1CCC(O)C1)=O)CC c1(CC)ccc(C=CC(N2CCCC2c2cn(-c3cnn(C)c3)nn2)=O)cc1 c1(C(=O)OC)ccc(NC(C2COCCN2C(C)=O)=O)cc1[N+](=O)[O-] N1(C(C)CC(N2CC3(C2)CN(C(=O)Cn2cnnc2)C3)=O)CCc2ccccc21 N1(C(C(CC#C)O)=O)CCC(C)(CNC(=O)C(c2ccc(C3CC3)cc2)O)CC1 C(=O)(CCS(C)=O)N(C1CCN(C(=O)C(C)C(C)O)C1)CC#C Cc1ccn2c(C(=O)N(C3CCCN(C(C4(CO)CCC4)=O)CC3)C)cnc2c1 c1(-c2nc(C3(C)CC(NC(COCC)C(=O)OCC)C3)on2)ccc(N)c(Cl)c1 c1(C(=O)NC(C2CN(C(Cc3nc(C)sc3)=O)C2)C)cc(F)c(F)c(Cl)c1F c1(CNC(c2cn(CC)nc2)=O)n[nH]c2c1CCC2 C(=O)(C1=CCCCC1C)NC1C(NC(c2snc(C)c2N)=O)CCC1 Cc1c(C(N2CCCC(C(C)NC(c3cn4c(n3)SCC4)=O)C2)=O)cccc1N c1(C(=O)NCCC(C)(C)NC(C2(c3cc[nH]n3)CC2)=O)cc(Cl)cc(Cl)c1F N1(C(Cn2c(C)ccn2)=O)CCC(C2CCN(C(=O)CC(C)C(F)(F)F)CC2)C1 Cc1ccncc1C=CC(=O)NC1CN(C(=O)CO)CCC1c1ccccc1 c1(NC)cc(C)cc(Cl)c1.n1(CCC)nnnc1CN(O)C=O c1(C(=O)NCCCCNC(C2C(C)(Br)C2)=O)ccc2c(c1)C(=O)OC2 c1(C(=O)CC2C3CN(N(C)NC(CCCC#C)=O)CC23)nccc2[nH]ccc12 CC1(C#CC(=O)NC2CCN(C(c3cc4n(n3)CCO4)=O)C23CC3)CCCO1 Cc1snnc1C(=O)NC(C1(O)CN(C(C2CCCCO2)=O)C1)C C(CC(C)C)(C(=O)NCC1CC2C=CC1C2)N(C(Cc1c(C)scc1)=O)C c1(C(=O)NCC2CCCC(CNC(c3n(C)ncc3Cl)=O)C2)cccc(F)c1N c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(Br)o2)=O)cncc(O)c1 Cc1ccc(C(N2CC(CCNC(=O)C#CC(C)C)C2)=O)c(C)c1Br C1(CNC(CC=C)=O)CC(C)N(C(=O)C=Cc2cc(C)no2)C1 C1(CCC(=O)CC2CC2)CCN(C(=O)CO)CC1.C1(OCC)CN(C(=O)CCO)C1 N1(C(C2N(CC)C(=O)CC2)=O)CC2CC(C1)N(C(C1CC(N(C)C)C1)=O)C2 c1(CC(N2CC(CCNC(C3(CCOCC)CCC3)=O)C2)=O)c(O)ncnc1O N1(C(c2c(CC)nco2)=O)CCCC(C2(NC(=O)CC3CCCCN3C)CC2)C1 N1(C(C2CC=C(C)CC2)=O)CCCC12CCN(C(c1cc(O)nc(C)n1)=O)C2 C1(C(N(CCN(C)C)Cc2nccs2)=O)(COC)CC2(CCC2)C1 Cn1ncc(S(C)(=N)=O)c1C(=O)NC12COCC(C(=O)O)(C1)C2 N1(C(c2c(CC)ocn2)=O)CCC(CCNC(=O)C(=O)NCCC(N)=O)CC1 Cc1cc(C(=O)NCC(O)CNC(=O)CC2CCSCC2)nn1C(C)C c1(OC)csc(C(N2CCC(CNC(c3ccnc(O)c3)=O)C23CC3)=O)c1OC c1(C(=O)NCC(CC)NC(=O)CCc2nncs2)ccc(F)c(Cl)c1 N1(C(CC(=C)C)=O)CC(NC(=O)CCc2ccc(CO)cc2)C2(CC2)C1 C1(CNC(C(CC)n2cncn2)=O)CC2(CC(NC(=O)CNC(=O)C3CC3)C2)C1 c1(C(N2CCC(NC(=O)Cc3cc[nH]c3)C(F)C2)=O)ccc2c(c1)S(=O)(=O)NC2 C(=O)(C1CCCc2cncn21)NC(C)CCN(C)C(c1cc(Cl)ccn1)=O c1(CC)cccnc1C(=O)NCC1(C)CCN(C(c2cc(C)nn2CC)=O)C1 O=S(=O)(c1cccnc1)N(Cc1cnc(N2CCOCC2)nc1)CC1CCCN1 N1(C(CC(COC)NC(=O)C(C)(C)SC)=O)CC2(CCC2(C)C)C1 c1(C(=O)O)cc(NCCc2ccc(Cl)cc2F)cc(S(=O)(=O)NCCO)c1 C1(C(C)C)CCC(C)(C)CC1.c12ccc(cc1)-c1cn(nn1)C2 N1(C(C(CC)(C)C(F)F)=O)CCC2(CC1)CN(C(=O)CCc1nnc(S)n1C)C2 C1(C(=O)OC)CCCN(C(=O)CC2CN(C(C3CN(C)CCO3)=O)CC2C)C1 c1(NC)ccc(C(N2CCC(NC(C3CCC3(F)F)=O)C(O)C2)=O)c(Cl)c1 Cc1cc(C(F)(F)C(=O)NCC(C)NC(=O)CCCC2CC2)cnc1Cl c1(C(=O)NC(C)CCCNC(=O)C(=O)N(C)C)cc2ccccc2cn1 C(=O)(CCCCC(N)=O)N(C1CCCN(C(=O)Cc2csc(C(C)(C)C)n2)C1)C C1(C(N2CC(COC)N(C(=O)CCc3ccoc3)CC2)=O)Cc2cccnc2C1 c1(C(=O)NCC2OCCCN(C(C=C(C)C)=O)C2)cnn2ccccc12 c1(CC(=O)NC(C)CCNC(=O)CC2CCC(O)C2)cc(Br)ccc1Cl C=CC(C)(O)CC(=O)NCC1CCN1C(C1CCCS1)=O N1(C(C(C)OCC)=O)CCCCC1c1nc(CCc2ccccc2F)nn1CC c1(C(=O)OCc2onc(CCOC)n2)cc2ccc(Cl)nc2s1 c1(C(N(CCCNC(=O)CCc2cnn(C)n2)C(C)C)=O)ccc(F)cn1 C1(NC(C2CCCC(F)C2)=O)C=CCN(C(c2ccc[n+]([O-])c2)=O)C1 N1(C(C2(COC)CC2)=O)CCCC(C2CCN(C(=O)Cc3nocc3C)CC2)C1 c1(C(N2CCC(C)(CNC(CC3(COC)CC3)=O)C2)=O)cc2c([nH]1)CCC(C)C2 c1(C(N2CC(N3C(=O)CC(NC(C(CC)F)=O)C3)C2)=O)ccccc1[N+](=O)[O-] N1(C(C(C)(C)OCC)=O)CCCC(CNC(=O)Cn2cc(COC)nn2)C1 CC(CCNC(C1CC(O)CCN1C(c1nn(C)cc1Cl)=O)=O)CC(C)(C)C c1(C(CNC(C)=O)NC(=O)C(Cl)=CCl)ccc(C)cc1 C(CC(C)CCNC(=O)CN1CCC(C)(C)C1)NC(C(C)C1CCC1)=O N1(C(c2cn(CCC)nn2)=O)CCCCC2C1CCCN2C(c1ccncc1)=O C1(NC(C2CCC(CC)CC2)=O)CCN(C(=O)C(C)CN2CCCC2)CC(O)C1 c1(C(N2CC3CN(C(C=C4CCC(C)C4)=O)CC3C2)=O)cccc2oc(O)nc12 C1(C(N2C(C3CCN(C(CCC=C)=O)CC3)CCCC2)=O)CC2CC1C1CC21 c1(C(N(CC(O)CNC(c2cc3c(s2)CCC3)=O)C)=O)nc(O)nc(O)c1F CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1ncc(Cl)cc1Cl)=O c1(C(=O)NC(C2(O)CN(C(CN(CCOC)C)=O)C2)C)cnc(O)cc1OC Cc1cc(F)c(OC(c2ccc(COC(c3cccs3)=O)s2)=O)cc1Cl c1(CC)ccc(Br)cc1C(=O)NCC(=O)N(c1nccs1)C c1(C(=O)NCC2(CNC(CS(N)(=O)=O)=O)CC2)cc2ccc(Br)cc2s1 Cc1nc(NCCOCF)cc(=NCc2noc3ccccc23)[nH]1 Cc1cc(C)n(C(C)C(=O)NC2(C3CCCN3C(=O)Cc3cncs3)CC2)n1 c1(OC)cccc(C(N2CC(CNC(=O)C(C3CC3)OC)C2)=O)c1F c1(CO)cccc(OC)c1O.c1(C(C)=O)ccc(NC(C2CCC(NC(C)=O)C2)=O)nc1 N1(C(CC(C(C)C)NC(=O)C(F)n2ccnc2)=O)CC(CO)C2(CCOCC2)C1 C1(CC(N2CC=CC(NC(c3c(C)nccn3)=O)C2)=O)CC(C)(C)CCO1 C1(NC(c2cc(F)ccc2C(F)(F)F)=O)CC2CCC(C1)N2C(C1CC1(F)F)=O C1(CNC(c2cnc(COC)s2)=O)CN(C(c2cn(C3CC3)nc2C)=O)CC1O C(=O)(C(C)S(C)(=O)=O)NCCN(CCC)C(c1ccc(CO)cn1)=O c1(C(CNC(C2COCCO2)=O)NC(Cc2nnc(C)o2)=O)ccc(F)cc1F C=CCC(CC(F)F)C(=O)N1CC2CN(C(=O)C3=CCCC(C)(C)C3)CC2(C)C1 C1(NC(c2c(C)nco2)=O)CC(NC(c2nc(Cl)ccc2Cl)=O)C12CCC2 c1(-c2nc(C(C(C(N3CCN(C(=O)OC)CC3)=O)C)C)on2)ccc(C)c(F)c1 S(=O)(=O)(c1cccc(C(=O)NCC23CCCC2CN(C(=O)C(C)(C)O)C3)c1)NC C#Cc1ccc(F)cc1C(=O)NC(C)CCNC(c1cc(C(C)C)ccc1F)=O C1(NC(C2C(C#N)CC2)=O)C2CCC(C2)C1C(=O)NC1CCCCC12CCC2 C1(C(=O)NC2CN(C(C(c3ccc(OC)nc3)(F)F)=O)C2)CCCC12CCC2 C=CCCN=C(NCc1ccc(C)cc1OC(C)C)NCC(C)(C)CC(F)F N1(C(c2n(C=C)ncc2)=O)CC2(CC2)CC1CNC(C1CC1c1ccn(C)n1)=O c1(SC)nc(NC2CN(C(c3cc(C(F)(F)F)nn3C)=O)CCO2)cc(O)n1 C1(Cn2ncc(NC(c3n(C(CC)C)nnn3)C3CC3)c2C)CCC(F)(F)CC1 CC1CCN(C(=O)C(=O)Nc2ccccc2)C1c1cn(C2C=CCCC2)nn1 N1(C(C2N(S(C)(=O)=O)CC2)=O)CCC2(C1)CN(C(c1ccc(O)nn1)=O)C2 CN1N=C(C(=O)NCC2(C(=O)NC3CCSC3)CC23CCC3)CCC1=O C=CCCC(C(=O)NC1CCOC(C)(CC)C1)NC(c1ccc(CC#N)cc1)=O c1(NS(CC2CCC(C)CO2)(=O)=O)ccc2c(c1)OCO2 c1(OC(C)(C)C)ccccc1CC(=O)NCC1CC(NC(C2(C)CC2F)=O)C1 N1(C(N(c2c(C)nsc2)C)=O)CCN(C)CC1c1ccccc1 c1(CC)ncccc1C(=O)NC1CCN(C(c2cc[nH]c2CC)=O)C1C1CC1 c1(CC(=O)NC2CC(N(C)C(c3ccc(OCCO)cc3)=O)C2)cc(F)cc(F)c1 C1(C(=O)NCCN(C(C(C)CN(C)C)=O)C)(COC)CC12CCC2 Cc1cn2nnc(C(N3CC(NC(C4C5C6CCC(C6)C45)=O)C3)=O)c2c(O)n1 c1(C(=O)NC(CCCNC(c2nn(CC)c(O)c2)=O)C)cc(S(C)(=O)=O)co1 C(=O)(CC(CC(C)C)NC(=O)Cn1cccn1)NC1CC(=C)C1 C1(NC(c2cc(C(=O)OCC)c(C)nn2)=O)CC2CCC1N(C(=O)CCSC)C2 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCC(CCNC(C1(OC(C)C)CCC1)=O)C C(=O)(C(CNC(c1ccsc1Cl)=O)N(C)C)N(C1CCN(C)C1)CCC C12(NC(=O)CCN3CCCCC3=O)CCC1CN(C(C1CCCCC1)=O)C2 C(=O)(C(F)CC(CC)CC)NC(CCCC)CNC(c1ccccc1F)=O C(=O)(C(C)(C)N=[N+]=[N-])NCCC1C(C)CN(C(c2cc(O)ncn2)=O)C1 C1(C(=O)NCC2(NC(CSc3n(C)cnn3)=O)CCCC2)CN=C2N=CNN2C1 c1(C(N(C(C)CCNC(=O)Cc2ccn(C)n2)C)=O)cc2c(nc1O)CCSC2 CC1CC(C)CN(CCOC2CC2)C1.C1(=O)C(O)CCn2cc(nn2)C2CCCN12 c1(-c2cn(C(C(=O)NCC(C)OC)C)nn2)ccccc1OC(F)F C1(CNC(C2CC2c2ccccc2)=O)CC(NC(C2(O)CCOCC2)=O)CC1O N1(C(CCCC(=C)C)=O)CC2CC(C)N(C(c3ccc(N(C)C)cc3)=O)C2C1 N1(C(c2ccc(CNC(C3N(C)CC3)=O)o2)=O)CC(CO)CC12CCC2 C1(C(N2CCC(C(C)C(=O)NCC=C(Cl)Cl)CC2)=O)CN(C)CCN1C CC1CCc2nc(Cl)nc(N3CC(CN(C)C(C4(C)CC4)=O)C3)c2C1 c1(CNC2CCCN(C(c3cc(C)cc(Br)c3F)=O)C2)c[nH]c2ccc(Cl)cc12 c1(OC)ccc(C(=O)NCC(C)N(C)C(c2cc(C)ccc2F)=O)n2nccc12 c1(C(N(C(C)CCNC(c2cc(C(F)(F)F)cs2)=O)C)=O)cccnc1F n1(CC(C)C)ccc(C(=O)N(C2CCCC2)CCNC(=O)C=Cc2ccsc2)n1 CC1(C#CC(=O)N2CCC(CF)(NC(=O)CC3CCSCC3)C2)CCCO1 c1(C(=O)NC(CNC(c2c(Cl)cnc(CC)n2)=O)C)ccc2c(c1)CCN(C)C2 C1(c2nnnn2CCCC2CC2)(NCc2ccn(C(C)(C)C)c2)CCC2CC12 N1(C(c2cnc(CC)[nH]2)=O)CCC(C2(NC(C3CC(C4CCC4)C3)=O)CC2)CC1 CC(=O)CCCC(=O)NC1(CF)CCN(C(c2cccnc2CO)=O)C1 C(=O)(CCCN(C)N=O)NCC(C)(C)OCCNC(C(CC=C)C)=O C(=O)(C1=C(CC)OCCS1)N1C(CCCC)CN(C(=O)C(F)C2CC2)CC1 C=CC(C(=O)NCCN(C(=O)C(O)C1CCC1)CCOC)NC(=O)OC(C)(C)C Cn1nccc1CCNC(c1cc(CNC(=O)C=CCN2CCCC2)no1)=O N1(C(CC(COC)COC)=O)CC2(C1)OC1(C)CC2(NC(=O)CC2CCCO2)C1 CC(CS(C)=O)C(=O)NCCC1CCN(C(C2CC=CC2)=O)CC1 c1(C(N2CCC(CNC(C3(C#N)CC4CC4C3)=O)CC2)=O)nnn2c1COCC2 N1(CC(C)C)CCC(C(N2CCCCC2CCCNC(C2CC(F)C2)=O)=O)CC1 N1(C(c2cc(C)cc(O)c2)=O)CCCC1C1CCCN1C(c1nccnc1C)=O c1(C(=O)NCC2CC(NC(c3cc(C)ncn3)=O)C2)ccc(N)c2ccncc12 N1(c2c(C#N)cncn2)CCOC2CN(C(=O)CCCc3ccccc3F)CC12 C(CC(C)(C)CC(=O)N(C(C)CN(C)C(C12CCC(CC1)C2)=O)C)OC c1(OC)ccc(CNC(=O)Cc2cnn(C)c2Cl)cc1 c1(C(=O)NCCN(c2snc(COC)n2)C2CC2)nsc2ccccc12 C(=O)(CCCC(C)=O)N1CC2C(CNC(c3c(CC)nc[nH]3)=O)(C2)C1 c1(C(=O)NC(C)(C(=O)NCCOC2CC=CC2)C2CCC2)ncn2c1CCC2 N1(CC)C(=O)NC(c2ccc(N)c(Br)n2)C2=C1C(C)(C)NC2=O N1(C(Cn2c(C)ccc2C)=O)CCC2CCN(C(c3ccn4ccsc34)=O)CC12 C=CCC(CC(C)C)C(=O)N1CCN(C(c2cccc(N)c2)=O)C(CCOC)C1 CCC(C(=O)NC(C)CNC(C1SCCS1)=O)SC C1(NC(COCP(C)(C)=O)=O)CN(C(=O)C(F)n2ccnc2)C2(CCCCC2)C1 c1(C(=O)NCC2COCCN(C(C(=O)N(C)C)=O)C2)cc2n(n1)CCNS2(=O)=O CC(C)C(CC(=O)N1CCCCCC1)NC(=O)C(CO)N(C)C O=C1NC(=O)C(CC(N2CCC(n3cc(CC(C(=O)O)C4CC4)nn3)CC2)=O)N1 CC1C2C(CCN2C(C2CC(C)(O)C2)=O)CN1C(=O)C1=COCC1 C1(C(=O)N(C(C)(C)C)C(=O)CN(c2ccccn2)CCN)CC2CCCCC2O1 C1(C(=O)NCC#CC)CCCN1C(=O)CC1CCSC1 N1(C(C(COC)O)=O)CCC(O)C(NC(c2ccc(-c3ccccc3)cn2)=O)C1 N1(C(c2ccsn2)=O)CCC2(CC1)CC(n1cc(CCO)nn1)CCO2 C(=O)(C(CC(C)C)N(C)C)NC1C(NC(C(OC)OC)=O)CCCC1 c1(OC)ccc(F)c(CN2C(C(=O)N(C)CCC3OCCO3)CC3CC23)c1F C(=O)(CCCCC(=O)N1CC(CO)(NC(=O)C(C)CC2CCCCC2)C1)OC CN1CC=C(CC(=O)N2CCC3CCC(C2)N3C(=O)CC(=O)OC(C)(C)C)CC1 N1(C(Cc2scc(C)c2)=O)CCCC(O)(CNC(=O)Cc2ccns2)C1 C(=O)(C1CCCc2sc(C)nc21)NC(CCOC)CNC(=O)COC1CCCC1 CC1CN(C(=O)Cc2ccc(F)cc2F)CCC1CNC(=O)C=CC(=O)N(C)C CON(CCC(=O)NCC=CCSC)C(=O)C(C)N1CCCC1=O C1(C(N2CC(OC)C(NC(=O)CC(Cl)Cl)CC2)=O)CC12CCC(=O)CC2 c1(OC)ccc(C(N2CCCC(CNC(=O)COCCF)C2)=O)nc1 c1(CNC(C2C(CC)NCC2)=O)cc(C)ccc1C C1(O)(CCC)CCN(C(C2CN(C)CCN2C(C2CCSC2)=O)=O)CC1 c1(C(=O)NCC2(O)CCN(C(CCC(=O)OCC)=O)C2)ccc(C)c(C)c1 c1(C(N(C)CC2CCOC2=O)=O)ncn2ccccc12.C12CN(C1)C(=O)CO2 C(=O)(C(C)CC(C)C)NCC1CN(C(c2c(CC)n(C)nc2)=O)CC1C c1(C(=O)NC(C2CC2(C)C)CC)ccc(CNC(c2cnc(CO)s2)=O)cn1 CC(CCN=c1[nH]c(N2CCOC(CC(N)=O)C2)nc2cc[nH]c12)C1CC1 C1(CC)C(C(=O)NC2CC3(CCCC3)C2)CCCN1C(=O)CCCOC N1(C(C2N(C(c3ccc(F)c(O)c3)=O)CCC(CC)C2)=O)CCOC2CCC12 C1(=O)N=C2NNc3ccc(cc32)N2CCC3(C(C(C)C)N1C3)CC2.C(=O)O C1(CC(=O)NCC2C(Cn3cc(CC=C)nn3)C2(F)F)CCC(OCC)CC1 c1(CN2C(C(N3CCCC3c3nn[nH]n3)=O)CCC2)cc(O)ccc1Cl CC(C)(CO)CCCNC(=O)CC1CCC(NC(C2(C#N)CCCOC2)=O)CC1 C1(C(=O)NC2CCC(NC(c3ccc(Cc4nccs4)o3)=O)C2)(CC)CCCC1 Cc1cc(C#N)ccc1C(=O)NC1(C(=O)NC2C(=O)OCC2CO)CC1(C)C N1(C(COC)=O)CC=CC(NC(c2ccn(CCF)n2)=O)C1 N1(C(C(COC)C)=O)CCCC(CCNC(c2cnn(C)c2C)=O)C1 N1(C(C(C)n2ccnn2)=O)CC2CCC1CN2C(=O)CC1CCN(C)CC1 N1(C(c2c(C)sc(Br)n2)=O)CCC(O)(CNC(=O)CC(C)C(F)F)CC1 c1(C(N2C3(CNC(C(C=C)(C)CC)=O)CC(C2)C3)=O)ccc(N)c([N+](=O)[O-])c1 C1(C)(CNC(C2(SCC)CC2)=O)CN(C(=O)CC2CCCOC2)CCO1 C12(NC(C(N3CCCCC3=O)C)=O)CC1CN(C(=O)CCc1cc[nH]n1)C2 C12(NC(c3cc(Cl)ccc3F)=O)CCN(C(c3conc3C3CC3)=O)CC1C2 N1(c2ncnc(NC(CCC)c3ccco3)c2C)CCCN(C)C(=O)C1 c1(C(c2ccc(C(F)(F)F)s2)N)ccc(F)cc1.C(CC(F)F)N(CC)CC N1(C(C(N(C)C(C2CC23CCC3)=O)C2CC2)=O)CCC(F)(F)CC1 c1(C(C(=O)NC(C)(CNC(=O)C=CCO)C2CC2)=O)ccc(F)cc1 Cc1[nH]c2ccccc2c1C(N1CCCC1C(=O)Nc1nnc(C2CCCC2)s1)=O C(CC1=CCN(C(=O)CC2CCCCC23CC3)CC1)NC(C1(C)CCC(=O)N1)=O CC(C)(C)C#CC(=O)N1CC2CC(C1)C2NC(c1ccc(C2CCC2)cc1)=O C1(O)(C(N(CCCNC(c2ccc(CCF)cc2)=O)C)=O)CC2CCC1C2 C1(C2CCN(C(=O)CCCC3CCC3)C2)(NC(=O)CCc2nncnc2O)CC1 c1(OC)ccc(Cl)c(C(=O)NCC(N2CCN(CCOC)CC2)=O)c1F c1(COC)nc(C)c(C(=O)NC2C=CC(CNC(c3cscc3SC)=O)C2)s1 C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NCC1(NC(C(C)OCCC#C)=O)CC1 C(=O)(C(O)CC(N)=O)N1CC2C(CNC(c3cc(C(C)(C)C)no3)=O)C2C1 N1(C(C(C2CC(NC(c3ccc(OC)nc3)=O)C2)F)=O)CC2(CCCCCC2)C1 c1(C2C(C(N(CCCNC(C3(NC(N)=O)CC3)=O)C)=O)CC2)c(Cl)cccc1Cl C=CCCCC(C(=O)OC)NCCc1cnc(OC)nc1 c1(C(N(CCS(C)(=O)=O)C)=O)ccnc(-n2cccn2)c1 N1(C(c2c(C)nncc2)=O)CC2CCC1C(CNC(C1(C)CCCS1)=O)C2 CCC(CC)C(F)C(=O)N1CCN(C(c2cccn(C)c2=O)=O)C(CO)C1 c1(CC)n[nH]c(=NCc2noc(C3CC3)c2C)o1 C(C(C(=O)NCC(O)C(=O)N(C)CC1CCCC1O)N(C)C)N(C)C c1(OC)ccc([N+](=O)[O-])cc1S(=O)(=O)NCCC1CC(C(=O)O)CN1 c1(C(=O)OC)n[nH]c(=Nc2cccc(F)c2NS(=O)(=O)Cc2cnn(C)c2C)o1 c1(C(=O)OC)cccc(CNC(=O)CCN2CCCC(C(N)=O)C2)c1O c1(CC)ncc(C(=O)NC(C)(CNC(=O)C(C)CSC)CC)c(C)n1 c1(C(CCC)C)nc(C)c(C(=O)NCCOc2nnc(C)s2)c(O)n1 N1(C(c2c(C)nc(C)o2)=O)CC(c2cn(CC3CC3)nn2)C(C)(C)C1 Cc1cc(-c2ccc(-n3cccn3)cc2)c2cc(-c3nn[nH]n3)ccc2n1 C1(NC(C(CC)OC2CCCCC2)=O)COC2(C1)CN(C(=O)CSC1CC1)C2 c1(N2CCCC(C)(C(N)=O)C2)ccc(S(=O)(=O)NCCC=CBr)cc1Br Cc1cn(C)nc1CNC(=O)NC1CC(c2ccccc2)C1 c1(NC(c2cccc(CN3CC(C(=O)OC)C3)c2)=O)ccc2c(c1)CCCC2 c1(C(N2CCC3(CC(OC)C3)C2)=O)cc2cc(Cl)cnc2o1 Cc1ccc(-c2ocnc2C(N2CCOC(CCN)C2)=O)cc1.C1(C=O)CCCO1 N1(C(C2CCC(C)O2)=O)CC2(C1)CN(C(=O)Cc1cn(CCO)nn1)CCO2 C(=O)(CCC(C)C#N)N1CC2C(C(=O)NCc3cncc(OC)n3)(C2)C1 c1(-c2cc(NCc3cccc(C(=O)O)c3)sc2)ccc(CO)c(F)c1F CS(=O)CCC(=O)NC(C)(C)CNC(c1cc(C2CCOCC2)[nH]n1)=O C1(NC(C2CC3(CCC3)CO2)=O)CC2(CCCN(C(C3CCCCC3)=O)C2)C1 c1(C(=O)NCC=CCNC(CC2C(C)(C)C(O)C2)=O)cc2ccc(O)cc2[nH]1 C1(Nc2cc(C)nc(N3CCC(c4coc(C)n4)CC3)n2)CCCCC(F)(F)C1 c1(C2CCN(c3ncnc(NCCC(C)(C)OC)c3C)C2)cccc([N+](=O)[O-])c1 Cc1n[nH]cc1CCNC(=O)NCC(C)(C)OC(C1(C)CC1)=O.C(N)=O c1(OC)cncnc1NC(C1CCN(C(=O)Cc2cncn2C)CC1)C C1(C(NNC(=O)C2OCC(C)C2)=O)CCCC(C)(C)CC1 C1(NC(c2c(N)nccn2)=O)CCC12CN(C(=O)C(c1cc(F)cc(Cl)c1)=O)C2 c1(C(=O)NCC2(OCC)CN(C(=O)C=Cc3ccccn3)C2)cc(C#N)c[nH]1 C1(C(N(CCCNC(CS(CC)=O)=O)C)=O)CCc2nc(C3CC3)ncc2C1 C(=O)(CC(C)C(C)(C)C)N1CC(NC(CCCOCCC)=O)C(n2ccnn2)C1 c1(C(=O)NC2CC3CN(C(CCN(C(C)=O)C)=O)CC32)cccc2ncnn12 C1(NC(c2c(C)nccc2)=O)CC2CCC1N2C(C1(C(C)(C)C)CCCCC1)=O c1(OC)cc(C(=O)NC2CN(C(=O)Cc3cccc(F)c3)CC2C#N)cnc1Cl C1(NC(c2cccc(OC)c2F)=O)CN(C(=O)CCC(C)O)CC2(CC2)C1 N1(C(c2c(C)n[nH]c2C)=O)CCC2(C1)CN(C(C13CCC(C1)C(C)O3)=O)C2 C(=O)(C(F)(CNC(C1COCCN1CC)=O)C(C)C)Nc1cncc(SCC)c1 C1(CCNC(C(C2N(C(Cn3ccc(C)c3)=O)CCC2)(C)C)=O)CCCCCC1 C(CS(=O)(=O)N1CCC(OCC2CCOC2)CC1)(C1CC1)OC C(N=c1[nH]c(=NCc2nnn(C)n2)[nH]c2cccnc12)C1CCn2c(C)nnc2C1 C12(C(N(CCC(C)NC(c3ccn(C(C)C)n3)=O)C)=O)C3C4C1C1C2C3C41C N(C1c2ccccc2CC1NC(=O)CC1CCC1)C(C(C)c1cc[nH]n1)=O c1(OC)ccc(Br)c(C(N2CCOC(CNC(=O)CC(O)C(C)C)C2)=O)c1 O=C(C1=COCCC1)NC1CCN(C(=O)CCOc2ccccc2)CC1F N1(C(c2c[nH]c(=N)o2)=O)CCN(C(C2CCCS2)=O)C(c2ccc(F)cc2)C1 C(=O)(C(C)(C)CNC(=O)Cn1nccn1)NC1C(OC)COC1 CC1CC(C)(C(=O)NCC23CC(NC(=O)CN4CC(C)(C)C4)(C2)C3)CC(C)O1 C1(Cc2nc(NC(=O)OC(C)(C)C)sc2)CCN(C(=O)CCc2ccco2)CC1 n1(C(C)C)nnc2c(NCCC3CCN(C(=O)C(C)CN(C)C)C3)ncnc12 C1(CC)CN(C(C2CC23CCOCC3)=O)CCC1NC(c1ccncc1F)=O n1(CC(=O)NCC)cc(CCN(C(C2CCCC2C)=O)CC)nn1 C12(CCCC1)C(=O)NC2.C1(C(=O)NCCC(=O)OCC)COC(CC)C1 CC1CCC(O)C(NC(=O)CC2CC(NC(=O)CC3CC(C4CC4)C3)C2(C)C)C1 C1(C(=O)NCCCCN(CC)CC)(CC)CCN(C(=O)C(C)c2ccsc2)C1 N1(C(COCCSC)=O)CCCC(CNC(C2(C)CCC(=O)N2)=O)CC1 C1(C2CC2)(C(=O)NCCCOCCNC(C=CC(CC)C)=O)CCOCC1 c1(C(N2CCC(OC)(CNC(C)=O)C2)=O)cc2c(Br)c(F)ccc2[nH]1 c1(OC)cccc(C(=O)NC2CC2C(=O)Nc2nc(Cl)ccc2I)c1C CC(C)C(F)(CNC(=O)CCc1cn(C)cn1)C(=O)NCC(F)F c1(CC)cc(C)nc(NC2(CO)CCN(C(=O)CC3CCOC(CC)C3)CC2)n1 C(CC1CC1)(C(=O)NC(CC1CCC1)C(=O)N1CC(OCCN(C)C)C1)OC c1(C(=O)NCCC(C)N(C(c2c(CC)ccs2)=O)C)ccc(C(C)C)c(C)c1 c1(C(N(CCN(C(CCC(=O)NC)=O)C)C)=O)nc(C(C)C)ncc1Cl CCS(=O)c1ccccc1C(=O)NCCOC1CN(C(=O)C(C)n2cncn2)C1 C(C(C(=O)NCCN(C(N)=O)C(C)C)NC(=O)Cn1nnnc1C(C)C)OC C1(C(=O)NNC(C2CC3CCCC(C2)N3)=O)CCOCC12CCC2 C(=O)(C1=C(C(F)Cl)N(CC2CC2)C(=O)NC1c1cc(I)c(F)cc1F)OCC C(C1CCOCC1)=CC(=O)NCC(CC=C)NC(c1cc(C)nn1CC)=O N1(C(c2n(C)nc(C)c2Br)=O)CCC(C)(C)C(NC(=O)CC(F)(F)F)C1 N1(C(c2c(C(N(CCC)CC)=O)ccs2)=O)CCCCCCC1 c1(OCC)ccc(CSC(C)C(N2CCCCC2CF)=O)cc1OC C1(C(=O)NC(CCC)CNC(=O)COC2CC=CC2)CCCCC1CC CCCC(CCCNC(=O)C(C1CCC1)OC)NC(=O)C=CC=C(Cl)Cl C(=O)(N=c1c(Br)c[nH]cc1Br)c1n(C)cc(N)n1.c1ccc([N+](=O)[O-])cc1 C1(NC(C2C(CNC(c3c(CC)n[nH]c3)=O)C2)=O)CCC12CCCC2 C#CC1(C(=O)OC(C)(C)C(C)NC(=O)OC(C)(C)C)CCC1 CC1CN(C(=O)C=CC2CC2)CC2(CCN(C(=O)CC3CCC(=O)C3)CC2)O1 C(CC1=CCN(C(c2ccc(Cl)s2)=O)CC1)NC(C1OCC(C)C1)=O c1(OC)cc(C)c(C(=O)NCCC2CCSC2)cc1OC N1(C(=O)OC(C)(C)C)CCc2cc(NC(N3CCOCC(O)C3)=O)ccc2C1 CN1CCC(NC(C2(CNC(C3OCCC3(C)C)=O)CCCC2)=O)CC1 N1(C(c2c(C)cc(C)[nH]2)=O)CCC2C(C1)CN2C(=O)CCN1C(=O)CCC1=O N1(C(C(CC)C)=O)CCc2ccccc2C(NC(C2Cc3ccncc3C2)=O)C1 CCC(CC)(C(=O)NC1CC(NC(=O)CN2CCCC2)C(O)C1)c1ccccc1 c1(CNC(=O)C2CC2)ccc(Cc2c(C(N3CCC(OCC)C3)=O)[nH]cc2)nc1 Cc1cn2cccc(C(=O)NC(C)CNC(=O)Cc3ccc4c(c3)OCO4)c2n1 c1(C(=O)NC2C(NC(CC3CCCN(C)C3)=O)C2)ccc2c(c1)OC(F)(F)O2 c1(Oc2ccc(C#N)cc2)ccc([N+](=O)[O-])c(C)c1.C(=O)(C(=O)NCC(OC)O)NCC N1(C(C2(CF)CCOCC2)=O)CCC2(CC1)CC(OCC)C2.C(=O)(C(C)C(C)C)N c1(CC(c2ccc(Br)cc2)C)nc(-c2ccoc2)nn1CC(F)F c1(OC)ccc(CC(C)C(=O)N(C)Cc2conc2C)cc1OC CC1(CNC(C2CC2c2cccs2)=O)CCCN(C(=O)Cc2ccc(N)cn2)C1 C#Cc1cnc(NC(C2CC23CCN(C(=O)CC2CCCC2)C3)=O)cn1 c1(C(C(=O)N(CC(=O)N(CC(=O)OCC)C(C)C)C2CCC2)C)ccn(C)c1 Cc1cc(C(F)(F)F)ncc1C(=O)NC1CC(NC(c2csc(Cl)c2)=O)C1 C1(NC(CS(C)(=O)=O)=O)CC2(C1)CN(C(=O)Cn1ncc(Br)n1)C2 C(CO)(CCCCNC(=O)C1CC1)NC(C1CCN(C)C1c1ccccc1)=O CCCCC(O)C(=O)N1CCC(CC(C)NC(c2cc(O)cc(O)c2)=O)CC1 c1(C(N2CCC(N(c3c(OC)n[nH]c3)C)CC2)=O)cc2n[nH]cc2cc1C C1(NC(C(CC=C)NC(=O)C=C(C)C(C)C)=O)CC2C=CCC(C1)C2 CCC(C)C(O)CC(=O)N1CC(CCNC(=O)CCC(=O)c2ccccc2N)C1 c1(C(=O)NC(c2ccccc2)CC)ccc(CN2CCOCC2)cc1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCN(C(COC2CCC(C)CC2)=O)CC1 c1(C(=O)NC2(CNC(C(CCC)(C)O)=O)CCOC2)ccc(C)c(OC)c1F C1(NC(C2(C)ON=C(C)C2)=O)CCC2CC1CN2C(=O)COc1ccccc1F N1(C(C2(C(=O)OC)CC2)=O)CCC(CCNC(C2CC2C(N)=O)=O)C1 c1(OCC)ncc(C(N2CC(NC(c3ccoc3)=O)C(O)C2)=O)cn1 C1(NC(C2(C)CC2Br)=O)CCC2(CC1)CC(NC(=O)COc1cccnc1)C2 Cn1nccc1C(C(=O)NC1(CF)CCC1)NC(C1CCC1O)=O C(=O)(CCC(C)(C)OC)N(CCCNC(c1cnc(CC)[nH]1)=O)CC CCCC(C(O)C(=O)N1CC(CO)CC(C)(C)C1)NC(=O)COC C1(C(=O)OC)Cc2ccccc2CN1C(=O)CNCC1CCC(F)(F)C(=O)N1 N1(C(CC=C)=O)CCC(C2CC(NC(=O)COc3cc(C)cc(C)c3)C2)CC1 C(=O)(C(F)CC(C)(C)NC(=O)C(F)n1ccnc1)NC(c1c(C)ncs1)C C1(CC)CN(C(C2COCCN2C(=O)CCn2ccnc2)=O)CC(=O)N1 C(=O)(C(C(C)(C)C)n1ccnn1)NC(CNC(c1c(C)onc1)=O)(C)CO N1(C(CN(CCC)C)=O)CCOC(CNC(c2sc(OC)nc2Cl)=O)C1 c1(-n2cc(CC3N(C(c4c(C)scc4)=O)CCC3)nn2)cc(O)nc(O)n1 c1(C(C)N)nc(CCN2CCCC2)nn1-c1cccc(OC)c1.CCCCOCCl C1(CNC(C(C)NC(C2C=CC=CC=C2)=O)=O)CC12CCCCC2 C(C)(C)(C(C)CC(=O)N(C(C)CN(C)C(C)=O)C)NC(c1c(C)cc(C)o1)=O C1(C(=O)NC2C(CNC(c3c(C)nco3)=O)CCC2)CCC(C(N)=O)N1C C12(C(=O)NCC(CNC(C3N(C)CC(F)C3)=O)(C)F)CCOC(C)(C1)C2 C=CC(C)(O)CC(=O)NCC(CC1CCCC1)C(=O)NCCC1CCOCC1 N#Cc1cc(F)ccc1C(=O)NC1CC(NC(=O)C=CC2CCOC2)C(O)C1 C12(C(=O)OC)CC(N)CC1CN(C(c1nnn3c1CCCC3)=O)C2 C(C(CC(C)C)NC(C1CC1C(C)(C)C)=O)NC(Cc1ccc(C)s1)=O C(CN=c1nc(N(C)Cc2ncccn2)c2c([nH]1)c(C)nn2C)c1ccc(C)s1 CC1CCNCCC1Cc1ccccn1.c1(N2C(=O)C=CC2=O)ccc(F)nc1 C(=O)(C#CC(C)(C)O)NC1CC(CNC(C(C(C)C)OC)=O)C1(C)C C1(CNC(C(C)N(C(=O)CCN2CCOC2=O)C2CC2)=O)CCOC1(C)C c1(C(=O)NC(CN(C(C2(C(C)C)CCC2)=O)C)C)csc2c1C(C)(C)CCC2 C(=O)(CS(=O)(=O)CCO)NCC1CCN(C(CC=CC)=O)C(C)C1 C(=O)(CC1COc2ccccc21)N1CCC(NC(c2c(C)scn2)=O)C1C(C)C C(=O)(C(C)(C)C(C)NC(C1CCC2(CC1)CC2)=O)N(CCC)C C1(CC(N2CC(OCCC(=O)NCC3C=CCC3)C2)=O)CCCCCCC1 C1(NC(C(C)(C)NC(CCCNC(=O)OC)=O)=O)CCCC2(CCC2)C1 C1(CCNC(C=C(C)C)=O)(NC(=O)Cc2cc[nH]n2)CCC1 c1(C(N2CCC(N(C(c3ccc(C(C)C)o3)=O)C)C2)=O)cc2occc2s1 C1(C(NOCCNC(Cc2cc(C)no2)=O)=O)CCCC(C)CC1.C(=O)C c1(C(=O)NC(C2CCCC2)CNC(C2CC2C(F)(F)F)=O)ncn2c1CCC2 C1(C2(N(C)C)CCC2)(NC(C2C3CN(C(C=Cc4n(C)ncc4)=O)C2C3)=O)CC1 c1(C(=O)NC2CC(N(C(C(C)SCCCC)=O)C)C2)cnn2c1OCC(C)(C)C2 O=C(C1=CS(=O)(=O)CCC1)NC1CCC(NC(=O)CC2CCC(O)C2)C1 C1(CNC(Cc2n(C)ncc2)=O)CC2CN(C(c3c[nH]nc3[N+](=O)[O-])=O)CC12 c1(C(N2CC(C)(OCC(=O)NCCOC3CCOC3(C)C)C2)=O)cncc(F)c1 CC1CC2(CC(C(=O)NC(CCF)C(=O)NCC3CCC=CO3)C2)C1 N1(C(C2(C(=O)OC)C3CCC23)=O)CCC(NC(=O)C(=O)NC(C)C)C1C(C)C N1(C(C2N(C(c3ccc(C#C)nc3)=O)CC(F)(F)C2)=O)CC2(CCOC(=O)N2)C1 c1(C(=O)NCCN(C(C2C(OC)CCC2)=O)CC2CC2)ccc(C)c(Br)c1 CC#CCCCC(=O)NC(CC(=O)NCCc1ncccc1F)C1CC1 C1(NC(Cc2cn(CC)nc2)=O)CN(C(=O)C(F)(F)C2CCCC2)CCC1CO c1(C(N2CCC(CNC(c3cnn(C)c3Cl)=O)C2)=O)cc(Cl)cc(F)c1N c1(NC(C(C2N(C(c3scc(C)c3)=O)CCC2)(C)C)=O)ccc(C)c(F)c1 c1(OCC(=O)NC(C)CC(C)NC(c2cc(C(N)=O)c[nH]2)=O)ccccc1C#N O=C1CN(C(=O)Cc2cn[nH]c2)C2CCN(C(C3CCCC3C(F)F)=O)CC2N1 C1(CNC(=O)CSC(F)F)CCCN1C(=O)Cc1nc[nH]n1 CCCC(CNC(=O)CC1CSCCO1)C(=O)N1CC(C)C1(C)C C1(CNC(c2sccc2Cl)=O)CNCCN1Cc1ccc(Br)cc1 CCC(C(=O)N1CC2CC(C1)CN(C(C1CC3(C1)CC1(CC1)C3)=O)C2)C(C)(C)CC c1(C(=O)NCC2N(C(C3(OC(C)=O)CC3)=O)CCC2)ccncc1Br C(=O)(C1CCCc2sccc21)N1CC(C)CN(C(c2ccnc(C)n2)=O)C(C)C1 C(=O)(CC#Cc1ccccc1)N1C(C)(CCC(=O)O)COCC1.S N1(C(CC2C=NN(C)C2=O)=O)CCCC(C2(NC(c3ccc[n+]([O-])c3)=O)CC2)C1 C1(C(C)C)CN(C(C23CCC(C2)C3)=O)CCN1C(=O)CN1CCNC(=O)C1 C1(NC(Cc2c(C)non2)=O)(CO)CCCN(C(C2(C)CCCC2)=O)C1 C(C(CC(C)C)C(=O)N1CCCC(C#N)C1)NC(C=CCOC)=O N1(C(c2c(C)onc2)=O)CC(C)C(NC(=O)CCC2CCC(=O)NC2)C(C)C1 n1(CCC)ncc(C(N2CCCC2CN(C)C(c2ccn(C3CC3)n2)=O)=O)c1Cl CC(F)(F)C(F)(F)CC(=O)NC1CCCC(CNC(=O)COCc2nc[nH]n2)C1 CC1(C)CCC(CNC(C2CC3CC3N2Cc2cnccc2Cl)=O)CC1 C(C(C(C)C(C)C)NC(c1nsnc1O)=O)NC(c1ccc(C)cc1)=O C1(OC)(CNC(=O)C(O)CSC)CCN(C(=O)CN(C)Cc2ccc(Cl)s2)C1 C#CCCCCC(=O)NCC1CCC(NC(C2(O)CCCC2)=O)C1 CCC(CC(=O)N1CCOCC1C(N1CCC(C)(C2CC2)C1)=O)C(F)F c1(C(=O)NCCN(C(C2CCN(C(C(C)C)=O)CC2)=O)C)ccc(O)c(F)c1F c1(OC)cc2c(cn1)N(C(=O)CNC1CC(C)OC1C)CC2 N1(C(=O)OC)CCCC(N=c2nc3c(ncn3C)c(NCCc3cc(Cl)no3)[nH]2)C1 c1(C(C)C)ncc2c(n1)CCN(C(c1cc(Br)cnc1-n1cccn1)=O)C2 N1(C(CCC=CC(C)C)=O)CCN(C(=O)C2=CCCCC2)CC1CC1CC1 C(=O)(C#CC1CCCC1)NC(CNC(C(CC(=O)OC)C)=O)C(F)(F)F c1(C(=O)NC2C3CN(C(CC(C)C4CC4)=O)C2C3)cc2nccnc2cc1F C(CCCC(=O)NCC(C1CCOC1)NC(C12CCC(C1)C2)=O)N(C)C CC1CCCC(C)N(C(=O)C(c2cn(C)nn2)NC(=O)CC2CC=CCC2)C1 N1(C(C(CC(C)C)=O)=O)CC2CCC1C(CNC(=O)Cn1cccn1)C2 C[S+](C)CCC(O)C(=O)NCC1(CC(=O)N(C(=O)CCC(N)=O)CC)CCCCC1 Cc1cccc(-c2ccc(C(=O)N(C)CCN(C)C(C3CCCCS3)=O)s2)c1 c1(C(N2CC(C)(NC(c3ccnc(N(C)C)n3)=O)C2)=O)ccc(F)cc1N C1(CC)CN(C(c2cc(CO)n(C)n2)=O)CCN1C(c1cc(OC)nc(C)c1)=O N(C(=NCc1ccnn1C)NCC1C(C)(C)C1(C)C)C(c1ncccc1F)C c1(C(=O)NC(C)Cn2cc(-c3ccc(C(=O)O)o3)nn2)nc(=N)cc[nH]1 c1(NCC2(C(C3CC3)NC(C=C(C)Cl)=O)CCCCC2)cc2occc2[nH]1 CN1N=C(C(=O)N2CCCC(O)(CNC(=O)CCCC(F)(F)CO)C2)CCC1=O c1(CN(C2CCCCCC2)CC(=O)OCC)c(Cl)cccc1Cl c1(N(C)CC2CCCN(C(C3C(C)(C)C3(C)C)=O)C2)ncnc2ccsc12 CC1CC(CNC(C2CC(C(F)(F)F)C2)=O)CCN1C(c1ccnn1C(F)F)=O Cc1cc(C(=O)N(CC(O)CNC(=O)CCOC2CC2)C)cc2c1CCC2 C1(CNC(c2c(C)occ2)=O)CCCC12CCN(C(C1(C(C)C)COC1)=O)CC2 c1(C(=O)NC2CC(C)(C)N(C(=O)CC#N)C2)occ2c1CCOC2 C1(NC(CCCC#C)=O)CC2CCC1N(C(=O)CCc1cnoc1)C2 c1(NC(C)=O)cc(C(=O)N(CCCNC(=O)C(F)(F)C(C)O)C2CC2)ccc1C c1(C(=O)OC)cc(=NCC(C)(C)C(C)NC(c2csnc2C)=O)[nH]c(Cl)n1 O=C(C1=C(Cl)CCOC1)NCCCC1CCN(C(C2COC(=O)C2)=O)CC1 Cn1ccc(C(=O)NCC=CCN(C)C2CC2)n1.C12COC(C1)NC(=O)CN2 CC1(C2CC2C(=O)NC2CCC(CC(=O)NCCc3nccs3)CC2)COC1 CCC(C)CCCCC(=O)N(C)CC=CC(=O)NC1CCCC12CC2 C=CCCCCCCC(=O)N(C1CN(C(=O)C(C2CCOCC2)C)CC1(C)C)C C1(CCCNC(C2CN(S(=O)(=O)C(F)(F)F)C2)=O)CCCCN1C(=O)CC1CC1 C(CCC(=O)NCC1CC1CNC(C1(C)CC12CC2)=O)N(C)C.C(COC)S C1(C(=O)NC(c2ncc[nH]2)C)CCN(C(=O)c2cc3n(n2)CCC3)O1 N1(C(CC2(OC)CC2)=O)CCC(C)(CNC(C2CN(C(C)=O)C2)=O)C1 Cc1cc(Br)cc(C(N2CC3(CCN3C(C3CCCO3)=O)C2)=O)c1F C=C=CC(C)C(=O)NC(C1(C(=O)NC(C)CO)CC1)C c1(CCC(=O)NCC2C(C(N(C3CCOC3)CC#C)=O)CC2)ccncn1 c1(C(N(C)C[Si](C)(C)C)C)cc(=O)n2nccc2[nH]1.C12CN(CC1c1nn[nH]n1)C2 C#CC1(C(N2CCC(NC(c3cc[nH]c(=N)n3)=O)C2)=O)CCCC1 Cc1nc(C(N2CCN(C(=O)C=Cc3ccc(O)cc3)CC2)=O)c2n1CCCC2 O=C(C(F)CC1CCCCC1)NC12CC(NC(C3CCC(=O)N3)=O)(C1)C2 C1(NC(CN2CCN(C(C(COC)(C)C)=O)CC2)=O)COCC(C)(C)C1 c1(C(N2C3C(NC(C(CC)CC4CCCC4)=O)C(C3)C2)=O)ccc(N)c(Cl)n1 C1(CNC(Cn2c(C)ncc2)=O)CCC12CCN(C(=O)C(C1CC1)C1CC1)CC2 c1(C(CC)NC(N2CCCC(N(C)C)CC2)=O)nc2ccccc2[nH]1 N1(C(C2(C)CC2)=O)CC2(C)CN(C(c3ccc4nsnc4c3)=O)CC2(C)C1 n1(CCCC(=O)NCC(=O)NCC(n2ccnn2)CC2CCCC2)ccccc1=O c1(C(=O)NC2C(CNC(C(C)N3CCC3)=O)C2)cc(Cl)cnn1 CC1C(NC(c2ccncc2C2CC2)=O)CC2CCC1N2C(=O)CC1CC1(Cl)Cl c1(C(N2CCC(C)(NC(CC(C=C)(C)O)=O)C2)=O)ccc(F)c(F)c1C c1(C(=O)NCCN(CCC)C(c2cc(CC)on2)=O)cnc2[nH]cnc2c1 Cc1nc(NCCC2CCN(C(C3CN(C(C)C)C3)=O)C2)c(C)c(C)n1 Cc1cc(-c2cn(CCNC(c3ccc(F)cc3Cl)=O)nn2)cnc1F c1(C(N2CC(NC(C3C(C(=O)OC)C3(C)C)=O)C2)=O)cn(C)nc1C CN1CCN(C(c2nc(=N)cc[nH]2)=O)C(C(=O)NC2(C)CC(N(C)C)C2)C1 C1(F)(C(=O)NC(c2ncnn2C)CC)CCCN(C(=O)C2=C(C)CC2)C1 CCC(CC(=O)NC(CNC(C1CCOCC1)=O)CO)C(C)C C(=O)(C#CC(C)(C)C)N1CC(OCCC(=O)NC(c2c(C)cccn2)C)C1 N1(C(CN(C(COC)=O)C)=O)CCC(CCN(C)C(C2NC(=O)CC2C)=O)CC1 N1(C(c2cc(CSC)on2)=O)CCCCC1CN(C(=O)C(Cl)=CCl)C C1(C(C(=O)NCCCC)N(CC)Cc2ccc(SC)cc2)CCOC1(C)C C1(NC(C2CCc3c[nH]nc3C2)=O)CC2CN(C(=O)CCn3cnnn3)CC2C1 C1(C(=O)NCCC(C)O)(CO)CCN(C(=O)CCc2ncccn2)C1 c1(C(=O)NCC2(F)CC(CNC(C=CSC)=O)C2)cnc2cc(O)ccc2c1 C1(NC(c2c(C)cc(N)cc2)=O)CCN(C(C2C(C)C2C)=O)CC12CCC2 CCC(C)(C)C(O)C(=O)NCCC1=CCN(C(=O)CCC2CCC(=O)NC2)CC1 C1(NC(CCCOCC)=O)CN(C(c2cnn3c2SCC3)=O)CC1(C)C c1(C(N2C(CNC(c3c[nH]c(=N)o3)=O)CCC(C)C2)=O)ccc2c(ccn2C)c1 c1(C(=O)NCCOCC)cc2c(-c3cc(OC)ncc3OC)cccc2s1 CN1C(=O)Cc2ccc(C(N3CCCCC(CNC(=O)C(O)C(F)F)C3)=O)cc21 CC1C2CCC(C2)C1C(=O)N(CC(C)(C)C(=O)NCc1cccnc1O)C CC1(C(=O)NC23CCCN(C(c4cc(Cl)no4)=O)CC2C3)CCCCNC1=O CCC1=NOC(C(=O)NOCc2nc[nH]n2)C1.c12ccc(s1)C(=O)NC2 c1(C(N2C(C(=O)OC)CCCC2)C(=O)NC(C)C)cc2cccc(OC)c2o1 CC(=O)CCCCC(=O)NCC(C)(O)CNC(c1csc(Cl)c1)=O N1(C(C2(C=C)CCC2)=O)CCCC(N(C)C(C2CCC(CCC)CC2)=O)C1 c1(OC)cccc(C(=O)NCC2CCCN(C(C3C(C)(C)OC3C)=O)CC2)c1C C1(CC)CN(C(c2ccc(C(N)=O)cn2)=O)CCN1C(=O)Cc1cncnc1O C12(C(=O)NC(CNC(=O)OC)C)CC(C)(CN1C(c1cncn(C)c1=O)=O)C2 C1(NC(CCOCC)=O)CCC(C)(C)CC1CNC(c1ccc(C2CC2)cn1)=O C1(C(=O)NC(CC=C)CNC(c2cc[nH]n2)=O)CCCCN1C(C)=O C1(CNC(C2C(CNC(=O)COCCF)C2)=O)CCCCCC1 CC1(C)CCN(C(=O)CC2CCSC2)C1CNC(C1CC(=O)NC(=O)C1)=O N1(C(C=CC=CCC)=O)CCCC(C)C1CO.c12cn(C)nc1CCNC2=O N12CCC(CC1(C)C)CNC2=O.C1(OCC)CC(C(C)NC(=O)CC)C1 CN1C(=O)CC(C(=O)NCc2ccc(Cl)nc2)C1C(=O)O Cc1c(C(N2CCCC(NC(C3(C)CCCN3C)=O)C2C)=O)cnc2ncnn12 c1(C(=O)NC(c2cccc(C)c2)C(=O)OCC)nc2n(c1C(C)C)CCCC2 CC1CCN(C(=O)COc2cccc(F)c2)CC1CNC(=O)Cc1cccs1 C1(CC)CN(C(c2ccc(OC)cc2)=O)CCC1NC(=O)C=CC(=O)NC1CC1 c1(CCC)nnc(CNCC(=O)OC(CC)OC)s1 c1(C(=O)NCC=CCNC(C2(C)CC2)=O)cn(CC(F)(F)F)nn1 Cc1cc(CCNC(C2(CF)CCN(C(=O)CCCC#N)C2)=O)nn1C N1(CCC(=O)NCC2CCN2C(=O)C(O)C2CC2)C(=O)c2ccccc2C1=O N1(C(CCN(C(=O)C(n2ccc(C)n2)C)CC)=O)CCCN(C)CC1C N1(C(c2c(C)noc2C2CC2)=O)CCCC2(CC(NC(=O)CSC3CC3)C2)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CCC(CNC(=O)COCC(F)F)C(F)(F)C1 N1(C(=O)Nc2cccc(-c3cc(C)c(O)c(N)c3)c2)Cc2cccc(Cl)c2C1 C=CC(CC)C(=O)NC1(CF)CN(C(=O)C(C)=C2CCC2)C1 c1(C(=O)NCC2N(C(Cc3c(C)noc3)=O)CCCC2)noc2ccc(Cl)cc12 N1(C(c2[nH]c(=NC)sc2)=O)CCC2CN(C(=O)CC3CC3(C)C)CC2C1 C(=O)(C(C)C(O)CCCC)NC(CCOC)CNC(=O)C=Cc1ccccc1 N1(C(CC2C(C)CCO2)=O)CCC2(C1)CN(C(=O)CCC1(C)CCC(=O)N1)C2 CN=c1cc(C(=O)NC2(C)CCCN(C(=O)Cc3ccco3)C2)c(Br)c[nH]1 c1(C(N2CC(CN3CCN(C(C4OCCO4)=O)CC3)C2)=O)c(F)cccc1Br C(=O)(C(C)(F)C(C)(C)F)N1CCCC(CN(C(C(CCC)NC(N)=O)=O)CC)C1 CC1CCN(Cc2ccc(-n3ccnc3)cc2)CCS1.C12CCCCN1C2=O Cc1cc(F)c(C(N2CC(NC(=O)CCCC(F)F)C(C)C2)=O)c(Cl)c1 C1(C2CC2)(CNC(c2ncc(C)nc2)=O)CCN(C(=O)CCCC2CC2)C1 C(=O)(C(C)CC(C)(C)C)NCC1(NC(CSCCC(C)C)=O)CCCCC1 Nc1cc(C(=O)NCC23COC(CNC(C4CC4(F)Cl)=O)(C2)C3)cc(F)c1 C1(NC(C2(CC)CCC2)=O)CCC2(CC1)CC2NC(c1cc(SC)no1)=O c1(OC)cccc(N2CCN(C(C3(c4ccccc4)CCNCC3)=O)CC2)c1 CCCC(CC(=O)OC)NC(=O)NCC(N1C(C)CCCC1C)c1ccccc1 C1(NC(CC2C(NC(C3(CN(C)C)CC3)=O)CCC2)=O)C2CCCOC12 CC(CS(C)(=O)=O)C(=O)NC1CCN(c2nc(Cl)ncc2F)C12CCC2 N1(c2[nH]nc(S(N)(=O)=O)n2)CCOCC2(COCC3CCCCN23)C1 Cc1nc(N2CC(CNC(C3CCCOCC3)=O)CC2C)cc(C(F)(F)F)n1 c1(CC(=O)NC(CCNC(C(CC)N(CC)CC)=O)C)c(Cl)cnn1C CC(C)CC(CNC(=O)NC1CC2CC2C1)C(=O)NC1C=C(C)CS1 N1(C(CC(=O)OC)=O)C2CCC1C(C(N1CCC(C)=C(F)C1)=O)C2 C1(CNC(CC2CCCN(C(C3CC(C)(C)C3)=O)C2)=O)CC2(CC2)C(=O)O1 C(CCCCC(=O)NCc1cccc(OCF)c1)N(C(C(C=C=C)C)=O)C C12CCC(C)CN1C2=O.c1(CC(C)=CC(N2CC3C=CC2CC3)=O)cc(C)c(N)cn1 C#Cc1cccc(CC(=O)NC(CCF)C(=O)NCCCOCC)c1 C=CCC(CC(F)F)C(=O)N1CCN(C(=O)C(C)n2cncn2)C2(CCC2)C1 c1(NC(C(C)N(CCC)C(c2ncccn2)=O)=O)cccc(F)c1O C1(NC(C2CC(C(=O)OCC)C2)=O)CC(C)N(C(c2ncncc2OC)=O)C1 c1(C(=O)NC2C(NC(c3[nH]nnc3C3CC3)=O)CCCC2)cccc2cc[nH]c12 c1(C(N2CC(CNC(C(C=C)O)=O)N(C)CC2)=O)cc(=O)n(C)c(=O)n1C N1(C(c2[nH]c(=N)sc2)=O)CCC(NC(c2ccc(CCF)cc2)=O)C(CO)CC1 c1(C(=O)NCC(C2CCC2)NC(C2CCCOCC2)=O)ccn2c1CCCC2 C1(C)(CC(=O)OC)CCN(C(=O)NC(c2ccc(Cl)c(Br)c2)C)CC1 CN1CC2(CCN(C(=O)Nc3ncccc3C(N)=O)CC2CO)C1 N1(C(c2cc(CNC(c3c(C)sc(O)n3)=O)sc2)=O)C(C)CC2CCCC12 N1(C(C2(OC)CCOC2)=O)CC2CCC(C1)N2C(=O)CC(CN(C)C)C(F)F C(C(=O)NCC=CCNC(C)=O)(c1cccs1)N(C(=O)OCC)C.C(C)(C)(C)O C1(C)(C(N(CCC(=O)NCCOC(C(=O)NCC)C)C)=O)CC(=O)N(C)C1 C1(C(=O)NCCC(=O)NCC2CCCCCC2)(CO)CCCCO1 C(=O)(C(O)C(F)(F)F)N1CCC(F)(CNC(C2CC(C(C)C)C2)=O)C1 C1(NC(c2occ(C)c2C)=O)CCN(C(=O)C(C2CC2)N(C)C)CC1CO c1ccc2cc[nH]c2n1.c12cccc(n1)CNC(=O)CC1CC(C1)C(=O)N2.CS N1(C23CC(=O)NC2CCCC3)CCCC2CN(C(=O)Cc3ccco3)CCC12 c1(COCCOCCOC)cc(NC(C2CC(O)C2)=O)ccc1Cl Cc1cnc(C(=O)NCC(C)NC(C2(C)CCNC(=O)C2)=O)cc1C N1(C(C(C)c2cc[nH]n2)=O)CCC2(C1)CN(C(=O)CCC(F)(F)F)CCO2 C1(NC(c2cnc(C)o2)=O)CCC2CN(C(C3CC(C(C)C)C3)=O)CC2C1 N1(C(CCOCCN(C)C)=O)CCC(CN(C)C(C23COC(C2)C3)=O)CC1 c1(C(=O)NC2CCN(C(=O)C(F)C3CC3)C2)cccc(OCC(F)F)c1 CC1CCCC(C)N1C(=O)NC1CN(C(C2CCCCCC2)=O)C1 C=CC1CCCCN1C(=O)C(CCF)NC(c1ccc(F)cc1C)=O C(=O)(N=S1(=O)CCC2(C1)OCCO2)C1(CC(CCCC)CC)CCC1 CCC1=C(C(=O)NCC(O)CNC(c2cc(C)c(F)cn2)=O)CCCO1 C1(C(=O)NC23CCCC2CN(C(C2CCCCO2)=O)C3)CCc2nnc(O)n2C1 N1(C(C2(COC)CN(C(=O)CN3CC4CC4C3)C2)=O)CC2CCC(C1)N2C C(=O)(C#CC1(C)CCCC1)NCc1ccc(CNC(C2CC(C(C)C)C2)=O)cc1 c1(C(=O)NCC2N(C(C3(C=C)CCC3)=O)CC2)cnc2[nH]ccc2n1 c1(C(N2CCN(CC(=O)OC)CC2)=O)cnc2n1CCOC2 Cc1ccc(C(=O)NC2CCC(CCC(=O)NCc3cscn3)C2)nc1 C1(NC(=O)C=CC2CCC2)CCCC(NC(c2cc(CF)on2)=O)CC1 CCCC(C)(O)C(=O)N1CC(F)(C(=O)NCc2cnn(C(C)C)c2)C1 CC1C(=O)N(C(c2cccc(F)c2)C2CCC2)CCC1=O N1(C(Cn2c(C(=O)OC)cnc2)=O)CCCC2(CNC(=O)C2)C1 c1(NC(N)=O)ccc(C#N)cc1[N+](=O)[O-].CC(C)CC1CNC(C(C)C)C(=O)N1 c1(OC)ncc(C)cc1NC(C1CC(C)(NC(c2ccc[nH]2)=O)C1)=O N(C(=NCCc1cccs1)N1CCC(N2CCCS2(=O)=O)C1)CCC1C(F)(F)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C(COCC)N=[N+]=[N-])C1)N1CCCCC(C#C)C1 c1(CC)c(C(=O)N(CC(C)O)CCNC(=O)CC2(C)CC2)cnn1C C12(NC(CN(S(N(C)C)(=O)=O)C)=O)CCCC1CN(C(C1CC13CCC3)=O)C2 CC1(C)CCCN(C(=O)CCc2cc[nH]n2)C1CNC(=O)C(F)C(F)(F)F C(=O)(CS(C)(=O)=O)NCC(CC)NC(=O)C(c1ccc(F)cc1)O n1(CCCOC)c(N2CCSCC2CC2CC2)nnc1-c1coc(C)n1 C12(NC(CNC(CC(C)C)=O)=O)CCCC1(F)CN(C(C1(C)CNC(=O)C1)=O)C2 c1(CCC(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)cnc2ccccn12 C1(C(=O)NCCC2(NC(CCCCCCC)=O)CCC2)CN2CCCCC2CO1 Cc1cc(=NC(=O)CC(O)C2CCCC(O)C2)[nH]n1C Cn1nnc(C(=O)NCC2CCC2NC(=O)C(O)Cn2cncn2)c1N c1(C(=O)OC)cccc2c1CCCC2NC(=O)NCCC1CC1C(F)F c1(OC)nc(C(=O)NCCCNC(C2(C)CC=CCC2)=O)sc1C C1(NC(=O)CNC(C2CCOCC2)=O)CC2CC(C1)N(C(C1CCCCO1)=O)C2 c1(NC(N(c2nccc(OC)n2)C2CCCNCC2)=O)cccc(Cl)c1F C(C(F)(CN=C(NC1CCC1)N1CCCC(C(C)C)C1)c1cccnc1)OCC C(=O)(C(C)CC(C)(F)F)NCC(CC)NC(c1ccc(C)c(Br)c1)=O C(=O)(C1(C)COc2ccccc21)NCC1C(C)(C)CCN(C(C2(O)CCC2)=O)C1 S(=O)(=O)(c1ccc(C#N)cc1)N(C(C1(C)N(C(C=COCC)=O)CC1)=O)CC CCCCC(O)C(=O)N1CC(C)(OC(C)=O)C1.C1(C)C(C)OC(=O)CN1 C=C(C)C(CC(=O)NCC1(F)CC(CNC(c2nc(Cl)sc2C)=O)C1)OCC Cc1cc(CN2CCCC(NC(=O)NC3CCC(C(F)(F)F)O3)CC2)cc(Br)c1 C1(C(N2C(CCC)CN(C(=O)CN3CCSCC3)CC2)=O)CCC2(CCCC2)C1 C1(C(=O)NCCC(=C)C)CCCCCC1NC(c1cc(C(C)C)[nH]n1)=O C1(CNC(C2(C=C)CC2)=O)CC2(C1)CN(C(=O)OC(C)(C)C)C2 C12(CNC(C3CCN(C(CN(CC)CC)C)CC3)=O)CCCC1OCC2 N1(C(C(C2CCC(F)(F)CC2)N)=O)CCCCCC1C=Cc1ccsc1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(c2cn(-c3c(C)ccc(Cl)c3)nn2)(O)C1 CC1CCC(Cl)=C(C(=O)NCCCNC(=O)CCC2CC2)C1 c12nc(C3CCC3)nn1C2c1ccccn1.n1(CC(n2nccn2)C)ccnc1 c1(C(c2ccon2)NCCCOC=C)nnnn1CC1CCCO1 N1(C(C2(NC(C)=O)CC2)=O)CCC2(CCC(NC(C3(O)CC(CF)C3)=O)CC2)C1 CCC(C)(O)C(=O)N1CCC(O)(CNC(=O)CCCc2cncs2)C1 CCCCCCCCC(C)C(=O)N1CCN(C(=O)Cc2nonc2C)CC1CC CN1CC(C(N2CCN(C(c3ncccc3-n3cccn3)=O)CC2)=O)CC1=O c1(C(N(C2CCN(C(C3CCCC(=O)O3)=O)CC2)CC)=O)ncccc1Cl CC(C)CC(C)C(=O)N1CCOCC1CN(C)C(c1cc(F)c[nH]1)=O O=[N+]([O-])c1cc(Cl)cc2c1OCCC2NCCC1CC2(CCC2)C1 C(=O)(C(C)(C)CC1CC1)NCC(CCNC(CN(C)C(=O)OC(C)(C)C)=O)O C1(C(C)NC(=O)Cc2csc(Br)c2)CCN(C(=O)C=CCF)CC1 c1(N(C(C2CC(SC)C2)=O)C)ccc(F)cc1.N12CCC1C(=O)O2 Cc1ccc(Cl)c(F)c1C(=O)NCC1CCN1C(C1CCC2CC12)=O c1(NC(C(CNC(C2CC(O)CN2C)=O)OC)=O)cc(C)c(F)cc1C c1(OC)ccc(C)c(OC)c1C(=O)NCC1CC(F)CN1C(=O)C1=CC(C)(C)C1 CC1CCN(CCC(=O)NCC2(O)CN(CCc3cccc(Cl)c3)C2)CC1 O(NC(=O)C(C)(C)C(C)(C)C)C(CC(C)C)C(=O)N(C)CC1CCC(=O)N1 c1(COC)nn(C)cc1C(=O)NCCC1(CNC(c2ccsc2Cl)=O)CC1 C1(CNCc2c(-c3ccc(F)cc3)n[nH]c2)COC2CCCC2O1 c1(NC(=O)NC(c2nncs2)C)n[nH]c(C(N)=O)n1 N1(C(C(C(C)C)OC)=O)CC2(C1)CN(C(=O)C(N1CCCCCC1)C)CC2CO N1(C(c2on(C)c(=O)c2)=O)CC(NC(c2cnn[nH]2)=O)CC12CCC2 c1(C(N2CCC(O)(CNC(C(C)C(F)(F)F)=O)C2)=O)c(N)cccc1[N+](=O)[O-] C(=O)(C(C1=C(C)C=CCC1(C)C)N(Cc1ccccc1C)CC1CC1)NCC=C N1(C(c2ccoc2Br)C)CC(NC(C2(C3CCCO3)CC2)=O)CCC1C c1(NC(C2(C(N3CC(=O)C(=O)CC3)=O)CC2)=O)cc(I)ccc1NC(=O)NC.CCO C(=O)(N=c1ccn(C2CC2)[nH]1)NC1C(c2c(C)n(C)nc2)N(C)C(=O)C1 N1(C(C2N(S(C)(=O)=O)CCC2)=O)CCC(O)C(NC(=O)CN2CCCCC2)C1 c1(C(=O)OC)cc(N2CCC(CNC(=O)C(CCO)N(C)C)C2)n2ncnc2n1 c1(C(=O)NCC2(C)CCCN(C(CCCCC#C)=O)C2)n[nH]c2ccc(Cl)cc12 c1(OCC)c(CN2CCOC(CCO)C2c2ccnn2C)cc(C)cc1C C1(C(=O)NCc2occ(C(=O)Nc3cnn(CC4CC4)c3)c2)CCCNC1=O C(CN=C(NCc1cncn1C)NC(c1ccccc1Cl)C(C)C)OCC C1(CC(=O)NCCOCCC#C)CCCN(C(=O)C(C)SC(C)C)CC1 C1(C(=O)NCCCN(C)C(c2ccccc2OC(F)F)=O)C2CCN1CC2 O=S1(=O)CC2CCCC2(NC(c2nnnn2C2CCC2)CC2CC2)C1 CCCCC(C(=O)NC1CCC(F)(CNC(c2csc(C)n2)=O)C1)C(C)C C(CCC(N)=O)(C(=O)N1CCC1(C)CC(C)C)n1cc(C(C)NCC)nn1.CCO N1(C(c2n(C)nc(C3CC3)c2)=O)CC2OCCN(C(=O)C3=CS(=O)(=O)CCC3)C2C1 C1(C(=O)NCC2(F)CC(CNC(c3nc[nH]n3)=O)C2)CCCCNC1=O N1(C(c2cc(OCC)n[nH]2)=O)CC(CNC(=O)COCCF)C(C)C1 c1(CC)ncc2c(n1)CCC(C(=O)NCC1CN(C(C3CC(O)C3)=O)CCO1)C2 N1(C(C(CNC(C2C(CC)OCC2)=O)CC(C)C)=O)CCC2(COC(=O)N2)C1 c1(CC(=O)N(C2CN(C(CC(C)(C)N(C)C)=O)C2)C)cccc2ncccc12 n1(CC(=O)N(CC(C)NC(=O)C(C)CSC)CC)cnc([N+](=O)[O-])n1 CCC(C)C(C(=O)NCCn1cc(CO)nn1)N(C)C(c1ccoc1)=O CC(C)(C)CCCCCC(=O)NC1CC1C1CCN(C(=O)C(O)CC(N)=O)CC1 N1(C(Cc2cc(C)ns2)=O)CCC(C2CCN(C(C34CCCC3C4)=O)CC2)CC1 N1(CC(=O)NCC2(C=C)CCC2)CCc2c(C(=O)OC)n[nH]c2C1 c1(NC2C(C)OCC2)ccc(Br)c(Cl)c1F CCCCCC(=O)NCCCNC(C1CC1c1cnn(C(C)C)c1)=O C1(C(=O)NC(C#CC)(C)C)CCCCN(C(=O)CCc2ccco2)C1 CCC(CC)CCC(=O)NCC(O)CCNC(c1cc(C#N)ccc1N)=O S(=O)(=O)(c1ccc2c(c1)OCCO2)N1CCCC(C(=O)NC(COC)C)C1 c1(NC(C2C(C)C2)=O)cc(NS(C)(=O)=O)cc(C#N)c1.c12csc(n1)NC(=O)C2 C12(CNC(COC(C)C)=O)CCC(CC1)N(C(=O)CC1CCCNC1=O)C2 C(=O)(C1=CCC(C)CC1)NCC1(OC)CCN(C(=O)Cn2nc(C)cc2C)CC1 C1(C(C)NC(=O)C(F)=C(C)C)CCN(C(=O)CC2(N(C)C)CC2)CC1 C1(C(=O)NC)COC2(CCN(S(=O)(=O)c3cc(C(=O)OC)sc3Br)CC2)C1 c1(C(=O)NCC(C)(C(C)C)NC(c2c(CC)c[nH]n2)=O)cc(F)ccc1C C1(C(=O)NCCN(C(=O)C=Cc2cccs2)C2CCC2)CCc2nnnn2CC1 C1(C)(C(=O)NCc2c(CNC(C3N(C(C)=O)CCC3)=O)occ2)CCCN1C c1(C(N2CCC(C(C)NC(c3c(C)ccn3C)=O)C2)=O)cnc2onc(C)c2c1 C(=O)(C(C)(C)CC(F)F)NCCCC(C)NC(C(C(C)C)C)=O C(CCCC(=O)NC1CCC1C(=O)NC(C)C(O)C(C)C)OC C1(C(N(CC(F)(F)F)CC)=O)CCCN(C(C2(F)CCOCC2)=O)C1 C1(NC(c2ccccc2)=O)CC2(C(=O)NCCc3ccc(O)nc3)COC1C2 CCC(C(=O)NCCCOCCC(N1CC=CC1(C)CO)=O)C(C)(C)CC C(CCC(C)(C)C(=O)NCC(CC(=O)N1CC(c2cc[nH]n2)C1)C1CCC1)OC C(C)(C)C(CNC(c1ncnc(O)c1F)=O)C(=O)N1CCN(C)CC1CCO CCC(C(=O)NCC1CC2(C1)CN(C(c1cc(F)ccc1C1CC1)=O)C2)C(C)C C(=O)(CC(C)NC(=O)C(C)CN(C)C(C1CC1C(=O)OC)=O)OC c1(NC(C(C2CC2)NC(C(C2CCCCC2)OC)=O)=O)cc(F)ccc1O CN(CCCC(=O)N1CC(NC(=O)CCc2ccc[nH]2)CC(C)(C)C1)N=O CN1CCC(c2ccccc2)(CNC(=O)Nc2cncnc2OC)C1.C1CC1 N1(C(C2CC(c3cn(C(CC)C)nn3)C2)=O)CC2(CCC(CCC(=O)NC)O2)C1 c1(C(N2C(CNC(C=COCC)=O)(COC)CCC2)=O)ccc(C)c(Cl)c1F C1(C2CCN(C(c3cscc3C)=O)C2)(NC(c2c(C)cc(C)s2)=O)CC1 c1(N(NC(=NC)NCC2CCN(S(C)(=O)=O)C2)CC)ccc(C)cc1.S(C)(=O)(=O)N CC1=NOC(C(=O)NC2CC(CNC(c3cncnc3C)=O)C2)C1C C1(CC)(NC(=O)CC(F)(F)F)CCCN(C(=O)COC)C1 Cc1oc(C(C)C)cc1C(=O)NC1CC(C)(NC(c2cccc(C(N)=O)n2)=O)C1 C1(C(N(CCCOCCN(C(=O)Cn2cccn2)C)C)=O)CCC12CCCO2 N1(C(C(CC(F)F)N(C(CCCCCC)=O)C)=O)CC2(CCC(=O)N2)C1 c1(C(=O)NC(CNC(COCC(C)C)=O)C(C)C)ccc2nc(C(F)F)[nH]c2c1 C1(C(=O)NCC(CC)NC(C2(CC)CCC2)=O)COCCOC1 N1(c2ccc(C(=O)OCC)cn2)CCC(C)C(NC(c2ccn(C)c2)=O)C1 c1(C(=O)NCC(CCCC)NC(=O)Cc2cc(C)no2)c(C)nc2sccn12 Cc1cn(C(C)C)cc1C(=O)NC1CC(CNC(=O)CCN2CCCCC2C)C1 Nc1cc(C(=O)NCCOCCNC(=O)CN2CCOCC2=O)cnc1N Cc1nn2c(c1CNC(=O)C(C)O)CN(C(=O)C(O)Cn1cncn1)CC2 N1(C(=O)OCC)CCC2(CC1)CN(C(C1(Nc3ccc(Cl)cc3O)CC1)=O)C2 C(C)(C)(CCCCNC(=O)CCC1CCCCC1)NC(C(CSC)C)=O C=CCC(C)(C)CC(=O)NC(C)(C)CN1CCN(C(=O)Cc2c[nH]nc2O)CC1 N1(C(CC(CC)O)=O)CCC2(CCN(C(=O)C=Cc3ccncn3)CC2)C1 C1(CNC(C(C)(C)SC)=O)N(C(=O)C(F)n2ccnc2)CCC1(C)C c1(-c2cn(C3CCCN(C(c4nc(C)oc4)=O)C3)nn2)cccc(Cl)c1Cl c1(CC)cc(Cl)ccc1C(=O)NC1CC(NC(C2CC(C(N)=O)C2)=O)C1 CN(OCC(F)(F)F)C(=O)C(Cc1cn[nH]c1)NC(C1CC12CC2)=O C1(C(=O)NCC2(F)CCC(NC(C3COC3)=O)C2)COc2cc(F)ccc2O1 C1(NC(CC2(NC(C3CCCN(C)C3)=O)CCC2)=O)CCCCNC1=O N1(C(C2C(C)C2)=O)C2CCC1CC(CNC(C1CC13CCOCC3)=O)C2 CC1=C(C(=O)N(C2CCCN(C(=O)CC3CCCNC3=O)C2)C)CCS1(=O)=O c1(C(N2CC=CC(C(=O)NC3CCCN(C)C3)C2)=O)cc(F)cc(F)c1 c1(C(=O)NC(C2N(C(C(CC)O)=O)CCC2)C)ccc(Cn2cccn2)cc1 CCC(C)C(=O)NCC(F)C(=O)N1CC(c2ccncc2)C1 N1(C(C(CC(=C)C)NC(C)=O)=O)CCCN(C(=O)Nc2cc(F)c[nH]2)CC1C N1(C(C(C)Cn2ccnc2)=O)CC2CC(C(N3CC(F)CC3C)=O)C(C2)C1 CC(C)CC(F)C(=O)NCCC1CCCCN1C(c1cc(-c2ccco2)[nH]n1)=O c1(NC2C(C)CN(C(C3(F)CCC3)=O)C2)ncnn2cccc12 c1(OC)ccc(-c2noc(C(N3CCCC(N4CCOC4)C3)=O)n2)cc1 c1(C(N(C2CN(C(CC(=O)OC)=O)CC2O)C)=O)cnn2c(Cl)cccc12 Cc1cc2c[nH]nc2cc1C(=O)N(C)CCOCCN(C)C(C1CC(F)C1)=O C(=O)(C1=CCC(C)(C)CC1)NC(C1CCCN(C(=O)CSCc2cscn2)C1)C CC1CC(=O)CCC1C(=O)NC(CCN1CCCC1)C(F)(F)F c1(NC(C2C(C(N(CC(c3ccccc3)C)C)=O)C2)=O)cnc(Br)cn1 c1(C(N2C(CNC(c3cccc(Cl)c3F)=O)CC(F)C2)=O)ccc2occc2c1 N1(CC=C)CCCN(C(=O)CCN(C(c2cc(SC)on2)=O)C2CC2)CC1 Cc1cc(C)c(CNC(C2(F)CCCC2)=O)c(C)c1.N12CCCC(C1)C2 C(=O)(CN1C(=O)CCCc2sccc21)NCC(CC)NC(C1(C)CC=CCO1)=O N1(C(C(=O)OCC)=O)CCCN(C(c2ccc(F)cc2C#N)=O)C(C)C1 N1(C(c2nc(CC)oc2C)=O)CC2CCC2(CCNC(=O)CCC#N)C1 C1(C(=O)NC2CC(Cn3cc(COC(C)C)nn3)C2)CN2CCC1(C)CC2 C1(NC(Cc2n(C)ncc2Cl)=O)CC(O)CN(C(c2cccc(CF)c2)=O)C1 c1(C(=O)NC2C(CC)CN(C(=O)CC3C=CCC3)CC2)ccc(S(C)=O)cc1 N12CCC3(CCC3NC(=O)CSCC1=O)CC2.CC(C)(C)OC(=O)NC=O c1(N(C(CC2C(NC)CCCC2)=O)C)ccccc1C(=O)O.N1(C(=O)C2CC2)CCCC1 c1(C(=O)NCC2CCC(NC(CCC(C)C)=O)CC2)ncn2cccnc12 c1(C(=O)NCC2(CC(=O)NCCO)CC2)cccc(CC#N)c1.c1(CS)ccc(Cl)s1 c1(OC)cc(Cl)ccc1C(=O)NC(C)(CNC(c1ccns1)=O)CC(C)C Cc1[nH]c2c(CNCC3OCCC3F)cccc2c1C c1(NC(=O)CCC(CNC(C(C)C2CCC2)=O)F)ccc(OCC#N)cc1 C(C1OCc2ccccc21)NC(c1nnc(-c2cccnc2)o1)=O CC1C(=O)CC1C(=O)NCC(C)N(C(=O)CCC1CCCOC1)C C1(C(=O)NC2COCC2O)CC2CCN(Cc3c(I)ccnc3F)CC12 C1(C(N2CC(OCC#C)C2)=O)CCC(C)(C)N(C(C2CCCN2C2CC2)=O)C1 C(=O)(C1SCCc2ccccc21)N(CCNC(C1COCCO1)=O)CC1CC1 C1(NC(=O)NCCNC(c2c(C)nsc2N2CCOCC2)=O)CN2CCC1CC2 C1(CC(=O)N(CC(=O)NC2CCCSC2)C)C(N(C)C)CC1O C1(OC)CC(NC(c2nnc(O)nc2O)=O)C12CCC2.C12CN(C1)C(=O)CO2 c1(CNC(C(c2ccnn2COC)N(CCC)CCC)=O)nnn(C)n1 Cc1cccc2c1ccn2CC(=O)NC1C=CCN(C(=O)C=CC(F)(F)F)C1 C1(C)(C(=O)NC(c2ccccc2F)CNC(C(CC)OC)=O)CC(F)(F)C1 C1(F)(CNC(C(C2CCOCC2)C)=O)CCN(C(c2c[nH]ccc2=O)=O)C1 N1(C(c2c(NC(=O)OC)cccc2)=O)CCC(F)(F)C(CNC(=O)CC(F)F)C1 N1(C(C2(CC)CCOC2)=O)CCN(C2CN(C(=O)C(=Cc3c[nH]cn3)F)C2)CC1 c1(Nc2cn(C3CCCN(C(C=C(C)Cl)=O)C3)nn2)ncnc(C)c1Br N1(C(=O)C=Cc2ccoc2)CCN(Cc2ccccn2)CC1C(F)(F)F N(C1CC2(CCCC2)Oc2ccccc21)C(=O)NC1(C(F)F)CCCC1 C1(NC(C2C(SCC)C2)=O)CC(F)(CO)C1.C(=O)C(CC)N(CC)CC Cc1cnc2ccccc2c1C(=O)NCCC(C)NC(=O)C(C)CF S(=O)(=O)(c1ccccc1Cl)NCCC(=O)NCCC1(NC(C2CCCO2)=O)CC1 C1(C(=O)NCCC2(NC(=O)CCc3ccc[nH]3)CC2)CC2(C1)C(F)(F)C21CCC1 c1(C(=O)NC(CC)CN2CCCC2)sccc1CNC(c1c[nH]c(=N)o1)=O CC1=NNC(=O)C1CC(=O)NC1CCC1.c12cc(ccn1)CC1CCCN1C2=O Cc1ccn2ncc(C(=O)NC(C)CC3CN(C(C4(C)CCCC4C)=O)C3)c2c1 C(C(=O)NC1(C(N2CC(F)(CO)C2)=O)CCCC1)(C(C)C)SC N1(C(=O)OC)CCCN(C(c2ccnc(-c3ccco3)c2)=O)CC1 CC(C)S(=O)(=O)C1CCN(C(C)C=O)C1.n1(CC2CNC2)cc(-c2cnn(C)c2)nn1 N1(C(C(c2ccn(C)n2)C)=O)CCC(C)(C)C1CNC(c1c(O)cncc1F)=O N1(CC(=O)NCCC(CNC(CC2C(C)C2)=O)(C)C)C(=O)c2ccccc2C1=O C1(C(N(CCNC(c2cccs2)=O)C2CC2)=O)CCCCS1.N12CC(C1)C2=O N1(C(CSC)=O)CCC(CNCCCCCc2ccccc2Cl)C(C)C1 c1(C(N2CC3(C(NC(C(CCC)OCC)=O)CC3)C2)=O)nc(O)nc(O)c1F C#CCCC(C(=O)OC)NC(=O)CCCCCBr C1(C2CN(C(C34CC(F)(C3)C4)=O)C2)(NC(c2cn(CC)nn2)=O)CC1 CC1=NOC(CC(=O)NC(CNC(=O)CCc2ccc(C)s2)CO)C1 c1(C(N(CCCNC(C2(C(F)F)CCC2)=O)C(C)C)=O)ccc(F)cc1Cl N1(C(C2(CCCC)CC2)=O)CC2(CCN(C(=O)CN3C(=O)NC(C)(C)C3=O)C2)C1 CC1CN(C)CCC1N(C)C(C1CC1C1CN(C(c2cccnn2)=O)C1)=O CC(C)(C(=O)N1CC(c2cn(-c3cc(OC(F)F)cc(F)c3)nn2)C1)S(C)(=O)=O C1(NC(=O)NCCOC2CCCO2)CCCN(C2CCCC2)C1 c1(C(=O)NCC(CC)NC(C2(F)CC2c2ccccc2)=O)ccc(OC)cc1 c1(C(N2CCC(O)(CNC(C(C)CF)=O)C2)=O)ccc(=O)n(CC(F)(F)F)c1 c1(C(=O)NCCC2CCN(C(C(C)n3cncn3)=O)C2)ncc(Br)cc1F C12(NC(C(CCCC)O)=O)CCC(CC1)N(C(c1cnnn1C1CC1)=O)C2 C(=O)(CCCC(C)(C)C)NCC1CN(C(C2(CC)CC=CC2)=O)CC1C(F)(F)F C#CCCC(C(=O)NC(C(=O)OC)C1(C)CC1)NC(C1C2CC3C(C2)C13)=O CN1CCN(C(c2cnns2)=O)CC1CNC(=O)C=CC(=O)NC1CCOCC1 N1(c2ncc(C(N3CCC(c4cccnc4)C3)=O)s2)CCS(=O)C2(CCC2)C1 O=S(=O)(c1ccc(NC(c2ccc(Cl)cn2)CO)c(F)c1)NC1CSC1 CC1CCNCCC1N(C(C1(C(F)(F)F)CC1)=O)CC1CCCCO1 C(=O)(C(C)(C)C(F)F)N(C1CCCN(C(c2nn(C)cc2Cl)=O)C1)C C1(N(C(=O)C(C)CSc2ccc(F)cc2)CC)CCN(CCC(=O)NC)CC1 C1(C(=O)NC2CC(n3cc(COC(C)C)nn3)C2)COc2cc(Cl)ccc2C1 c1(C(N2CCC(NC(=O)COc3ccsn3)CC2)=O)ncnc2ccsc12 C1(F)(C(=O)NCCCCC)CC(NC=O)C1.C1(CC(=O)N)CC(F)(F)C1 C1(C(=O)Nc2cccc(NC(=O)COc3ccsc3Cl)c2)CCC2(CCC2)CO1 N1(c2cc(NCC(C)F)nc(COC)n2)CCn2c(nn(C)c2=O)C1 c1(C(N(CCCCCC)CCNC(=O)C(CO)C(C)(C)C)=O)nccc2ncncc12 c1(C(N2CC3C(NC(CCC=CC)=O)(C3)C2)=O)cnc2ccsc2c1 c1(C(=O)NC2CCCN(C(C(CC)C(C)(F)F)=O)CC2)oc2ccccc2c1C C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)C(C)C)CC2(CC2)C1 C=CCCCC(C(=O)NC1(C)CC1(C)C)NC(=O)Cc1c(C)noc1C c1(C(=O)NCc2cc(SC)oc2)nc(C(=O)NCCOC2CCC2)c(C)o1 c1(OC)cc(C(=O)N(CC(O)CNC(=O)Cn2ncn(C)c2=O)C)cnn1 c1(C(=O)NCC#CCNC(C2CCC(C)(CC)O2)=O)cc2ccccc2nc1O CCCCCCCC(=O)NCC1COCC1NC(c1ccc(Br)o1)=O c1(C2C(C(=O)NCC(C)C)C2)ccncc1-c1cnc(-c2ccccc2)s1 CCCCC(C)CCC(=O)N1CCC(NC(c2cccc(N(C)C)c2)=O)CC1C C1(C(=O)NC2C(NC(C3CSC3)=O)COCC2)Cc2nnsc2S1 C(CNC(=O)Cn1cc(CO)nn1)(CC(=O)N(C)C(c1ccsc1)C)OC CN1C(=O)CCCC1C(=O)NC(C(=O)NCc1cnc(N(C)C)nc1)C1CC1 c1(OC)cccnc1CC(=O)NCCCN(CCCNC(=O)CCOC)C C12(NC(c3c(C)nc(C(C)OCC)s3)=O)CCCC1N(C(C1(SC)CC1)=O)CC2 c1(C(=O)O)ccoc1C(N1CC(=C(F)CNC(C2C(C)C2)=O)C1)=O C1(C(=O)NC2(CC(=O)NCCCCCCF)CCC2)CCCC(F)C1 C1(CCOC)CN(C(c2cccc(C(F)F)c2)=O)CCN1C(=O)C1=NOC(C)C1 c1(C(=O)NC2CN(Cc3ccnc(O)c3)CC2F)cn2ccc(Cl)cc2n1 CCCCC(CNC(c1cncc(-n2cccn2)n1)=O)NC(=O)C(C)N1CCC1 C(=O)(C1Cc2ccccc21)NCCN(C(c1cncc(OC)c1)=O)C1CC1 c1(SC)cc(C(N2CCC(O)(CNC(c3ccc(F)o3)=O)C2)=O)ccc1F O(NC(=O)C(c1ccco1)NC(c1c[nH]c(=NC)o1)=O)C(CC)C Cc1cc(Br)ncc1NC(C1CCN(C(c2ccc(F)cc2)C)C1=O)=O Cc1cnc(NC(c2cscn2)C)c(S(=O)(=O)NC(CO)C2CC2)c1 N#CC1(C(=O)NC2CCC(NC(=O)CCn3cccc3)CC2)CCOC1 C(C)(CNC(=O)CN1CCCC1C)(CC(C)C)NC(CCc1ccc(C)o1)=O C1(CNC(CC2C(C(=O)OC)C2)=O)CCN(C(=O)CC2(NC(C)=O)CCCC2)C1 c1(C(=O)NCC(CNC(=O)Cc2ncc(Br)s2)OC)cnc(O)n1C C(C(C)(C)CC(=O)NCCC1CC(NC(c2ccc(Cl)nc2OC)=O)C1)OC Cc1ccc(C(F)(F)C(=O)NC2CC(NC(c3ncncc3Br)=O)C2)cc1 N1(C(CC(=O)NC)=O)CCCN(C(c2ncnc(OC)c2OC)=O)C(C)C1 C12(NC(COCCC)=O)CCCC1N(C(=O)Cn1cc(C)cn1)CCC2 c1(-n2cc(C3(C)CCCC3)nn2)cccc(C(=O)NCCc2cccnc2F)c1 C(CC(C(=O)N1CCC(C#N)C1)NC(=O)CCCOC)OCC C1(NC(N2CC(C(=O)OCC)CC2(C)C)=O)CCC2(CC1)CC(CN(C)C)C2 S(=O)(=O)(c1c[nH]ccc1=NCC1(F)CC(CO)C1)NC(C)C(C)CO CCC(CN(C)C)CC(=O)NCC1C(C(=O)Nc2cc(C)cnc2O)C1(C)C c1(OCCC)ccc(C(=O)NCC(C)CN(C(=O)C(C)C#N)C)cc1 N1(C(COC(C)C)=O)CC2(C1)CN(C(=O)CNC(c1cccnc1)=O)C2 C1(CNC(c2cc(C(F)(F)F)on2)=O)CN(C(=O)C(F)F)CC1C(F)(F)F CCC1(CC)CN(C)C(=O)OC1.C1(OC)CC(=O)N(C(C)C2CC2)C1 c1(C(=O)NCCN(C(=O)CCN(C)C(C)=O)CCOC)cn(C)cc1C C(CCCCC(=O)NCC(c1cn[nH]c1)NC(=O)Cc1ccc(F)c(F)c1)OC N1(C(=O)NCc2ccc(SCC)o2)Cc2c(OCCOC)ccc(F)c2C1 N1(C(CCN(C)CC)=O)CCC2(CC1)CCN(C(=O)CC1CCC(C)O1)C2 c1(C(=O)OC)c(C(=O)NCC(C2CCOC2)NC(C2CCCCC2)=O)n[nH]c1C C(=O)(C1=C(F)CN(C(C2Cc3nccn3C2)=O)CC1)NCC1C(C(C)C)C1 C1(CNC(C2(CCC=C)CC2)=O)CC2CC(C1)N(C(c1cnn(C)n1)=O)C2 C1(CC)(NC(=O)CC2(O)CCC2)CCCN(C(=O)C(C)CC2CCCC2)C1 C(=O)(C(C(C)C(C)(C)C)N1CCC2CC(C(=O)NC)C2C1)NCCCCCC C(=O)(CCCCC(C)C)NC(C(C)NC(c1n(CC)cc(Br)c1)=O)C C(=O)(C(CCCOC)NC(c1c[nH]c(C(N)=O)c1)=O)NCC=C c1(NC2C(C(F)(F)F)CCN(C(C(CC=C)C)=O)C2)nc(C)c(C#N)cc1Cl c1(N2Cc3c(nc(C)s3)C2)nc(=NC(C)C2CSC2)nc(-c2ccncc2)[nH]1 c1(C(N2CCC(C)(CC(=O)NCC(c3ccco3)O)C2)=O)cc2occc2[nH]1 O=C1NC(Cc2ccc(F)c(Cl)c2)C(=O)N1Cc1cccc(-n2cncn2)c1 C(=O)(C(C)CC(C)C(C)=O)NCCOCC(=O)NCC(=O)OCC(=C)C CCC(C(=O)NCc1cc(C(=O)N(C)CC2CCCN2C)cs1)N(C)C N1(C(N(CC(=O)OCC)C)=O)CCC(O)C(C(=O)NC(C)C)C1 c1(C(=O)NCCNC(=O)NCCc2ccncc2)ccc(C2CC2)cn1 c1(C(=O)NCC2N(C(C(C(CC)O)C)=O)CCC2)c(Cl)ccc(C)c1O c1(OC)ccc2c(Nc3cc(-c4ccc(OCC)cc4F)ccn3)ncnc2c1 C1(C(=O)Nc2c(C)cccc2F)CC2CCCCC2N1C(c1nc(Cl)sc1Cl)=O c1(C(=O)NC2CN(C(CCC=C)=O)C(C)C2)c(Br)c(C)nn1C C1(C(N2C(C)(CCO)CC2)=O)CC2(CCN1C(c1cccs1)=O)CC2 N1(C(c2cc(C)[nH]n2)=O)CCC(NC(c2ccc(OC(F)F)cc2)=O)CC1C CC(C)CCCC(=O)NCCC1CN(C(=O)CCCn2ccnc2)CC(C)O1 C1(C2CN(C(=O)CCCCn3ccnn3)C2)(NC(c2c(C(N)=O)csc2)=O)CC1 C(=O)(C(C(C)(C)C)C1CCCC1)NCC(CNC(CCN1CCC(C)CC1)=O)F c1(OC)ncc(Cl)cc1C(N1CCOC(CCCNC(=O)C(CSC)OC)C1)=O C=C(C)CC(C(=O)NCC(C)(C)CC)NC(c1oc(C)nc1C)=O c1(OCC(N2CC(CS(N)(=O)=O)C2)=O)ccc([N+](=O)[O-])c(F)c1 C1(N(C(COCCOCC)=O)C)CCCC1NC(=O)Cn1cc(C(C)F)nn1 C1(NC(C(CC=C)NC(C)=O)=O)CC2CN(C(=O)C(C)(C)C(=C)Cl)CC2C1 N1(c2cc(CCC)nc(Cl)n2)CCC(NC(c2nsc(OC)n2)=O)C(CO)CC1 C1(C(=O)NC2C(NC(Cc3c(C)non3)=O)CCC2)Cc2ccccc2S1(=O)=O c1(C(N2CCC(NC(CC3(C)CCC3)=O)C2)=O)cccc2ncsc12 N1(C(CCSCCCC)=O)CCC(C)C(NC(=O)CCCCCN(C)C)C1 c1(N2CCC(CCC)C2)nc(=NCCc2nccc(O)n2)[nH]c2c(F)cccc12 c1(C(=O)OC)cccc2c1CCC2NC(=O)Nc1c(I)ccnc1OC c1(OC)cc(=NCC2CN(C(=O)CCOCC(F)(F)F)CC23COC3)[nH]cc1C C1(NC(Cn2nc(C)oc2=O)=O)CN(C(c2ncccn2)=O)CC1C1CC1 c1(OC)cncc(C(N2CCC2CSCC)=O)c1.c12cc(c(C)s1)C(C)NC2=O CC1(NC(=O)CSC2CCC2)CCN(C(c2cc(Cc3nncs3)on2)=O)CC1 c1(C(=O)NCC2C(NC(CC=CC(C)(C)C)=O)C2)cnc2ccccn12 c1(C(N(C2CCC(NC(C3(COC)CCCC3)=O)C2)C)=O)ccc(P(C)(C)=O)o1 C(=O)(CCC(C(=O)O)NC(c1ccc(F)cc1C(F)(F)F)=O)N(C)C C(=O)(C(=O)C(C)(C)CC)N1CC(C(=O)NC2(CC=C)CCOC2)OCC1 Cc1cn(C)cc1C(=O)NC(C)(C)CCCNC(c1ncc[nH]c1=O)=O C12(CNC(C(C)(C3CC3)OC)=O)CCC(CC1)N2C(C1CN(C(N)=O)C1)=O C1(CNC(C2(CC)COC2)=O)(CO)CCCN(C(=O)CC2CCCC2O)C1 c1(C(C)=O)cc(O)cc(C(=O)NNC(=O)c2cncnc2)c1O C1(N(C)C(=O)NCCC(=O)Nc2ccccn2)COC(=O)C1 c1(CC)ccc(C(=O)NC2CCN(C(=O)C(C)CNCC)C2C2CC2)cc1Cl Cc1cccc2c(C(=O)NCCN(C)C(c3cnc(Cl)c4ccsc34)=O)cnn12 C1(CNc2cc(N(C)CC3CC(F)(F)C3)ncn2)CCCC1S(C)(=O)=O C(=O)(C(C(C)O)N(C)C)NCC1(OC)CN(C(c2cc(C3CC3)[nH]n2)=O)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CC(NC(=O)C(C)C2CC2)Cc2ccccc21 N1(C(C2C(C(=O)Nc3nccc(F)c3F)C2)=O)CCc2ccc(Cl)cc2C1 N1(C(c2ccc(C)s2)=O)CCC(NC(c2cn(C)cn2)=O)C(C)C1 c1(C(N(CCOC)CCNC(=O)CC2CCOC2=O)=O)cc2ccccc2o1 N1(c2ncnc(C)c2F)CC(NC(=O)CSCCN(C)C)C2CCCCC12 C1(NC(=O)CC2CCOC2)CC2(C1)CC(NC(C1CC13CCCCC3)=O)C2 C1(NCC(N2CCC(F)(F)CC2)=O)CCCCC2CN(c3nnco3)CC12 C1(C(=O)NC(C(=O)NCC)C)CSCCN1C(=O)CCN1CCCC1 c1(SC)ccccc1C(=O)NC1CCOCC1NC(=O)CCCn1ccnc1 CC1CCC(CC(=O)NCCC(=O)NC2CC3CC3C2)OC1 CCC(C)C(O)C(=O)NCCCC(C)NC(c1c(OC)nsc1OC)=O c1(OC)n[nH]c(C(N2CC(CNC(=O)C=Cc3cn(C)cn3)CC2C)=O)c1Cl Cc1nc(C(=O)NC2CCCC(N(C(=O)CCCc3ccsc3)C)C2)n(C)n1 C(C(=O)NCCN1CC(c2cncn2C)(c2nccn2C)C1)(C(C)C)S.CO N1(CC(C(CCCCC)=O)=O)CCC(C2CCN(C(=O)C(C)=C3CCCC3)C2)C1 N1(C(C=C(C)c2ccco2)=O)CC(CNC(c2coc(CC3CC3)n2)=O)C(C)(C)C1 CC1=NN(C)C(=O)C1CC(=O)NCC1CCCC(CNC(C2CC=CCC2)=O)C1 N1(C(C(C)CC(N)=O)=O)CCC(CNc2nccc(S(C)(=O)=O)n2)C(F)(F)CC1 N1(C(c2c(Br)c(C)n(C)n2)=O)CC(CNC(=O)CC(C)(C)O)CC(C)(C)C1 C1(C(=O)NCC(CNC(COCC=C)=O)C(F)(F)F)CCn2ncnc2C1 CS(C)(=O)=NC(=O)C(=O)NC1CN(C(=O)COc2cccc(CO)c2)CC1F c1(CCCC(N2C(COC)CN(C(C)=O)CC2)=O)ccc([N+](=O)[O-])cc1O c1(OC)ccc(C(C)N(C)C(C2CC2CC(=O)Nc2cn(C)nc2C)=O)cc1 N1(C(c2ccc(C(C)(C)C)s2)=O)CC(NC(C2CCCO2)=O)CC(O)C1 c1(CC)ccccc1N(C(=O)CCOCCCNC(C1CC(=O)N(C)C1)=O)C Cc1ccc(F)cc1CC(=O)NC1CN(C(=O)C(O)c2ccsc2)CC1C N1(C(CC(=O)NCC#C)=O)CCC(C)N(C(=O)C(C)Cn2ccnc2)CC1 c1(SCCC)ccc(C(=O)NC2CCCCC2NC(=O)CNC(=O)C2CC2)cc1 c1(CCC(=O)NCc2cccc(CN(CCOC)C)c2)ccc(C)cc1C N1(C(C(C(=O)OCC)F)=O)CCCC(NC(=O)C(C(C)CC)N(C)C(C)=O)CC1 c1(C2C(OC)C2)ccc(-c2nnc(-c3cccc(-n4cncn4)c3)o2)cc1 C1(COC(N2CCCC(C(=O)OCC(F)(F)F)C2)=O)CCCC(F)(F)C1 c1(C(=O)OCCCCCCC)cc(Cl)cc(S(=O)(=O)NC)c1F C(=O)(C1=Cc2ccccc2OC1)N1CC2N(C(C3CCC(=C)CC3)=O)C(CC2)C1 C(=O)(CC(C)(C)C)NC(C)C(=O)NCC1CC1NC(=O)Cc1cncc(Br)c1 CC1(C)COC(C(=O)NC(CNC(c2ccccc2OCCF)=O)C2CC2)C1 C(=O)(C1=NOC(CN)C1)N1CCC(CN(C)C(c2ccc(N=[N+]=[N-])cc2)=O)C1 CCCCC(c1nnnn1CCOC)NCc1cccn1CC C1(NC(c2ccc(C)s2)=O)C2CC3CN(C(C4CC(C)N(C)C4)=O)C1C3C2 C(=O)(C(F)(F)C(O)C1CC1)NCC1N(C(c2ccc(C(C)C)cc2)=O)CC(F)C1 C1(CC(=O)N(CCC(=O)NCCOCCOC(F)F)C)CC2C=CC1C2.C(C)N CC(C)(C)CCC(=O)NCC1(NC(C2CCC(C3CC3)C2)=O)CC1 Cc1cn2c(n1)CCC(C(=O)NCC1CN(C(=O)CCOC3CC3)CC13CC3)C2 c1(CC(=O)NC23C(CCN(C(c4[nH]c(=N)sc4)=O)C2)C3)ccc(F)c(Cl)c1F C(C(=O)NC(C)CC(N)=O)(C(C)(C)C)NC(C=Cc1c(C)n[nH]c1)=O C1(NC(C(=O)NCC=C)=O)CCN(C(C2CSC(CC(=O)OC)C2)=O)CC1OC C#Cc1ccccc1C(N1CC2CN(Cc3ccn(C4CCOCC4)n3)C2C1)=O C1(NC(CSCC(C)OC)=O)CN(C(C2CN(C(N)=O)C2)=O)C2(CCC2)C1 CC1(C)CC(C(=O)N(C2CCCC2)CCNC(c2ccn(CCF)n2)=O)C(=O)O1 C1(NC(CCN(C)CC)=O)CCCC1C(N1CCC(CCO)C1)=O c1(C(=O)NC2CCCCN(C(C3(C)CCCO3)=O)C2)cccn2nncc12 C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1CN(C(C(CC)N(C)C)=O)CC1C c1(C(=O)NC2CC(CNC(C3CC4(CSC4)C3)=O)C2)[nH]c2ccccc2c1Cl c1(C(=O)NCC2CC3CC3N2C(c2cccc(CF)c2)=O)cc2cccn2cn1 C1(C)(C(N(CC(CC)C)C)=O)CCN(C(C2CCOC2)=O)CC1 CCCCCC(C(=O)NC12CC(CNC(c3ccsc3Cl)=O)(C1)OC2C)C(C)C c1(OC)cc2[nH]c(=NC(C(F)F)c3cccc(F)c3)[nH]c2cc1OC C1(NC(c2cc(C)sn2)=O)C2CCC(C2)C1C(N1CCC(NC(=O)C2CC2)C1)=O Cc1cncc(S(=O)(=O)NCc2cc3cnccc3[nH]2)c1 c1(C(N2CCOCC(NC(C(C(C)C)C3CCC3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(C(CN(C)C(=O)C2CC2)O)=O)CCCC(N(S(C)(=O)=O)C)C1 C#Cc1ccc(C(=O)NCC2(OC)CCN(C(c3c(Cl)noc3C)=O)C2)nc1 C(=O)(CC(C)CCC(=O)Nc1cnn2c1OCC(O)C2)OC(C)(C)C c1(OC)ccc(N)c(C(N2CC3(CC3)CC2CNC(c2cscc2OC)=O)=O)c1 Cc1cnc(C(=O)NCCOC2CN(C(C3(C)CCCCC3C)=O)C2)cc1C#N c1(C(=O)NC(c2cn(-c3cccc(F)c3F)nn2)C)ncc(Cl)cc1Cl C(CN=c1[nH]c(=N)[nH]c(=NC2CC3(CC3)C2)[nH]1)N(C(C)C)C1CC1 N1(C(C(C=CCCC)O)=O)CCC2(CC(NC(c3ccc(Cl)c(O)c3)=O)C2)C1 Cc1ccc2[nH]c(C(=O)NCC3(F)CN(C(c4ccc(Cl)s4)=O)C3)cc2c1F N1(C(CC(C)C)=O)CC2CCC2(C(=O)NC(C2CC3CCC2C3)C)C1 C1(F)(CNC(CC2(C=C)CC2)=O)CCC(NC(c2cncn2C)=O)C1 O=C(C1=Cc2c(ccc3ccccc23)OC1)NC1CCC2(CC1)CN(C(=O)C1CC1)C2 N1(C(C2(NC(CCCOC(C)=O)=O)CCC(C)(C)C2)=O)CCC(=O)N(C)CC1 C(C(C)(C)CCCC(=O)NCC(CC(C)C)NC(=O)CS(C)(=O)=O)SC Fc1cc(Cl)ccc1CNC(c1nnnn1CCO)c1ccno1.c1(C)ccccc1 C1(NC(c2c(CCC)nco2)=O)CCN(C(=O)CCn2ccccc2=O)C1(C)C c1(CC(=O)NCCC2CCCN2C(=O)C(O)C(F)F)ccc(F)cc1 C1(NC(c2c(COC)cc[nH]2)=O)CCN(C(=O)C(C)=C2CC2)CC1F Cc1cc(Cl)c(O)c(NC(c2nnnn2C)CCc2ccsc2)c1F N1(C(=O)Nc2scc(SCC=C)n2)CCc2cc(C(=O)OC)cnc2C1 c1(C(N2CCC(C)(C)C(CNC(c3cn[nH]c3)=O)C2)=O)cnc2ccnn2c1N CC1CCCC1(F)F.c1(C(C2(c3ccon3)CCC2)N)nnnn1C1COC1 c1(C(N2CCCC(C(O)C(F)(F)F)C2)=O)cnccc1C(F)F C(CCCC(CO)NC(=O)C(c1ccccc1)N(C)C)NC(c1scc(C)c1)=O Cc1noc(C)c1C(N1CCC(CCNC(C2CCC(C(N)=O)O2)=O)C1)=O c1(C(N(CCCNC(C2CC23CC3(F)F)=O)CC)=O)nccc2ccsc12 c1(COC(C(=O)NCC(CNC(C=CCCC)=O)C)C)ccncc1 C1(NC(=O)NC2CC(C)CC(C)C2)CC2CC3(CC2C1)OCC(C)(C)CO3 C(C(CC1CC1)C(=O)N(C)CCOCC1CC1)NC(C(C)SC)=O C(CCCCC(=O)N1CCC(NC(=O)C2=COCCO2)CC1)NC(N)=O N1(n2cc(CCCS(N)(=O)=O)nn2)CCN(CCCF)CC(O)C1 C1(NC(C)=O)CCCCC1.C(C(=O)N(CCCNC(=O)CO)CCO)C1CCCO1 C1(NC(COC(C)C)=O)CC2CC1CN(C(=O)CCc1cccc(N(C)C)c1)C2 C(=O)(CCCC(F)(F)CO)NC1CCC(N(C(C(C)(O)C2CC2)=O)CCO)CC1 c1(C(N(C(C)C)CCN(C)C(C2COC(=O)O2)=O)=O)cc(F)cc2nn[nH]c12 C(CC(C(=O)N(C)Cc1ccc(F)cc1)NC(C1CCCC1OC)=O)OCC c1(N(C)C)cc(C(=O)NC2(CO)CN(C(C3COC(C)(C)C3)=O)C2)cc(Cl)n1 C1(CNC(c2n[nH]c(C)c2C)=O)CC(C)CN(C(=O)C=CC2CCOC2)C1 C[Si]1(C)CCC(CNC(C2CC(N)C2)=O)C1 N1(C(C(C)C2CCOC2)=O)CC(NC(=O)CCF)C(N=[N+]=[N-])C1 C(=O)(C1CCCn2nccc21)NCC1CCCN(C(CCCCCSC)=O)C1 CCC(CNC(c1nc(=N)[nH][nH]1)=O)(CC)C(=O)NCCC1CCC(=O)N1 C(=O)(C(=O)C(C)(C)C)NC(CCNC(C(C)SC(C)C)=O)(C)C C1(CC)CCCN(C(=O)CC(C)CC)C1C(=O)N(C)CC1COCCO1 Cn1nc(C(=O)NC2CCC(NC(=O)NC3CC3)C2)c2ccccc12 C(=O)(C(F)(F)C(O)CC)NCCCCCN(C(c1nc(CC)sc1)=O)C(C)C CC1(C)CC2(CC(NC(=O)NCCC3=CCCCC3)C2)C1 c1(N(C(c2cccc(Br)c2)C(=O)NCCCF)CC)ccc(F)c(C)c1 N1(C(C(C)SCC)=O)CCOC2(CCC(NC(c3cc(C)cnc3C)=O)CC2)C1 C(=O)(CC(C)CC(C)C)NCCCN(C(c1c(C(C)C)cccc1F)=O)C N1(C(CCc2nnc(CCC)o2)=O)CC=C(CNC(c2conc2C)=O)CC1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1C(C)(C)CCC(n2cc(C3(C)CC3)nn2)C1 N1(C(COCC=C)=O)CC2(C1)CN(C(c1ccc(-c3ccncc3)o1)=O)C2 N1(C(c2cc(SC)c(C)o2)=O)CCC(C)(C)C1CNC(C1(O)CCCCCC1)=O C1(NC(c2ccc(C#C)o2)=O)CC2CCC(C1)N2C(=O)CCCCC(C)C C(=O)(C1=CC2CCC(C1)C2)N1C(C(=O)NCC(C)CC(F)(F)F)CCCC1 CCC(C)C(C(=O)NCCCC1(NC(c2cnn(C)c2N)=O)CC1)NC(N)=O c1(OC)ccc(CC(=O)NC(CCN(C)C(C23CCC2CC3)=O)C(C)C)cc1F N1(C(C2(C#C)CN(C(=O)CCCCC)C2)=O)CC2(CCC2)C12CCC2 C(C(O)CC(F)(F)F)NC(C1C2(CC(NC(c3c(OCC)scc3)=O)C2)C1)=O c1(C(N(C(C)CNC(c2cnc(O)c(F)c2)=O)C)=O)cccc(S(=O)(=O)CF)c1 c1(C(N2C(C)CN(C(C3CCSCC3)=O)CCC2)=O)cc2c(nn1)CCCC2 c1(C(=O)NCC(=C2CN(C(CC3CCCN(C)C3)=O)C2)F)cc2cccnn2n1 c1(CNC(C(=O)NCC2CCC(C)C2)=O)ccc(Cl)cc1 c1(CC(=O)NC2(C)CC(NC(COCC(=O)OC)=O)C2)nc2c([nH]1)CCCC2 c1(C(N2CCC(NC(c3nn(C)c(O)c3)=O)C(F)C2)=O)ccc(I)c([N+](=O)[O-])c1 C1(CC(=O)NCC=CC(N2C(C=C)CC2)=O)CC2(CC2)CO1 N1(C(C2(CC=C)CCCCC2)=O)CC(NC(=O)CN(C)C2CC2)C2(CC2)C1 c1(CC(N2C3CC(CN(C(C(C)(C)C(F)F)=O)C3)C2)=O)cc(Cl)ccc1[N+](=O)[O-] C1(C)(C(=O)NCC(C)(C2CC2)NC(CCc2c(C)noc2C)=O)CCCNC1=O Cc1nc2cccc(C(N3CCCNCC3c3ccccc3)=O)n2n1 N1(C(c2ccc(C(C)C)s2)=O)CCC2(CC1)CC(CNC(C1COC(=O)N1)=O)C2 N#Cc1ccc(C(N2CCCCC2C(N)=O)=O)cc1Cl.c1(O)cccc(CO)c1 CCC(CC)C(C)C(=O)N1CCCC(CC)(NC(c2cn(C3COC3)nn2)=O)C1 N1(C(CCOCC#C)=O)CC2=C(C1)CN(C(c1occc1COCC)=O)C2 c1(C2(C(=O)NC3CC(NC(C4(CO)CC4)=O)C3)CC2)ccc(OC(F)F)nc1 N1(C(c2n(CC)nc(C)c2)=O)CC2CC1CN2C(=O)COc1c(C)cccc1Br c1(N(CC(C)NC(C2COCC(C)(C)O2)=O)C)ccnc2ncnn12 c1(C(=O)NC2(CNC(c3ccc(CC#N)cc3)=O)CC2)cc(Cl)cc(Cl)c1O c1(C(N2CC(n3cc(NC(CS(N)(=O)=O)=O)nn3)C2)=O)cccc2c1CCN2 C1(C)(CNC(C=NOC)=O)COCCN(C(=O)CC2(C)CCCC2)C1 C(=O)(CC(C)C(=O)NCC(C)CNC(c1ccnc(N(C)C)c1)=O)OCC N1(C(C2C(C=C)OCCC2)=O)C2CCC1CC(CNC(=O)COCCN(C)C)C2 C1(C)(C(N2CCCC(CCOC)C2)=O)CN(C(=O)C(=O)NOC)C(C)(C)C1 C(N=c1[nH]c(=NC(C)c2ncnn2C)c2[nH]ccc2[nH]1)c1ccc(CC)nc1 Cc1noc(C)c1C(c1nnnn1C)Nc1cccc(CC2CC(=O)NC2=O)c1 Nc1ccccc1C(=O)NCc1cn(CCCC(=O)NC2CCCC2CF)nn1 C1(NC(Cc2n(C)ccc2)=O)CCC(C)(CNC(c2ccc(C(F)F)nc2)=O)C1 c1(C(=O)NCCCC2N(C(C3CC(N(C)CC)C3)=O)CCC2)cc(Cl)ccc1F C=CC(C)CC(=O)NC(CO)C(C)NC(=O)C(C)OC O=C1CCCC(C(N2CCC2CNC(=O)CC2COCC2O)=O)CC1 C1(CN(C(=O)NC(C)CC(O)c2ccccc2)CCO)CCN(c2cccnc2)CC1 c1(C(=O)NCC(CNC(CCOC)=O)CO)cc(C)cc(OC)c1O N1(C(C(CC=C)OC)=O)CC2CN(C(C3(NC(C)=O)CCCC3)=O)CC2C1 C(=O)(C1=CCCOCC1)N(C(C)C)CCN(C)C(C1CC(=O)C1C(C)(C)C)=O N1(C(C2CCN(C)CC2)=O)CC2CN(C(c3cc(C4CC4)no3)=O)CC2(C)C1 N1(C(C=C(COC)C)=O)CC(NC(C2CCC3(CCC3)CC2)=O)CC12CCCC2 N1(C(CSC2C(=O)OCC2)=O)Cc2ccccc2C(NC(c2cn[nH]c2)=O)C1 N1(C(CONC(=O)CCC2CCC2)=O)CCc2n[nH]cc2C1 CCCCC(CC)CC(=O)NC1(C)CCCCC1C(=O)NC(CN(C)C)CO c1(CC)cccc(C(N2CCOCC(CNC(c3ncncc3F)=O)C2)=O)c1N Cc1cc(C(=O)NCCOCCn2cc(CC3CCCCC3)nn2)co1 CCN=C(NCc1ccnn1C1CCCCC1)NC1Cc2ccccc21 Cc1nc[nH]c(=NCC2CN(c3nc(C4CC4)cs3)C2)c1Br C1(F)(C(=O)NC2CN(C(=O)Cn3cc(C(N4CCOCC4)=O)nn3)C2)CC=CCC1 C1(C(=O)NCCCOCC#C)CCC2(CC2)N1C(=O)C(C)S(N)(=O)=O C1(CNC(C(=C)F)=O)CCN(C(c2ccc(Br)cc2CC#N)=O)CC1O CCCC(C(=O)NCc1ncoc1C1CN(C(c2ccn(C)c2)=O)C1)OC C1(CC)(NC(=O)C=CCO)CCCN(C(=O)C(c2ccccc2)n2cncn2)C1 C1(C(=O)NC2C(OC)COCC2)CC12CCN(C(c1ccn(C(F)F)n1)=O)CC2 c1(C(=O)NC2CCC(NC(=O)COc3cccnc3)CC2)cnn2ccncc12 CC(CSc1ccccc1)C(=O)N1CCC(N(C(=O)CNC(N)=O)C)C1 C1(CNC(c2c(CC)nccn2)=O)CC2(CCN(C(c3cncs3)=O)CC2)C1 C1(NC(CC(C)C)=O)CC(CNC(C2C3CCC2CC3)=O)C12CCC2 C(=O)(C(O)C(F)(F)F)N(CC(CN(C(c1cccc(OCC)c1)=O)C)O)C c1(CC)ccc(CNc2ccc(-c3ccc(C)nc3C)cc2)c(C#N)c1 c1(-c2nc(-c3cc(OCC)ncc3)nn2-c2cccnc2)ccc(CC)nc1C c1(COC2C(O)CN(c3nccc(-n4ccnc4)n3)C2)ccc(I)c(Cl)c1 c1(C(=O)NC(C(C)NC(C(CCOC)C)=O)(C)C)ccc2[nH]c(=N)n(C)c2c1 N1(C(CCC=C(C)C)=O)CC(NC(C2CC(C)(C)CO2)=O)CC1(C)C N1(C(C(C)C)=O)CCC(O)(C2CCN(C(C3CN4CCN3CC4C)=O)CC2)C1 Cn1ncc2c1CCCC2CNC(=O)CNc1c[nH]nc1C1CCNC1 N1(C(C(C)OC)=O)CC2CN(C(c3cc(-c4ccccc4Cl)[nH]n3)=O)CC2C1 C1(C(N(C(C(=O)OC)C)C)=O)CC1C1CN(C(=O)CC2OCCOC2C)C1 c1(C(N2CC(CNC(c3ccnc(OC)n3)=O)C2)=O)n[nH]c2c1CC1CC21 N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CC2CCN(C(=O)CC3(O)CCC3)CC12 c1(C(=O)NC(CC=C)CNC(=O)CCc2nc(C)no2)cc(C)c(F)cn1 C1(CNC(C(C)C2CC2)=O)CN(C(=O)CC2CCC(F)(F)CC2)CCC1(F)F Cc1cc(C(N2CC(F)(CNC(C34CC(C)C3C4)=O)C2)=O)nc(O)n1 C1(OC)CCCCC1CN1CCOC(c2ccc(OC(F)F)cc2)C1 C(C(C)(C(=O)N1CCN(CCNC(=O)COc2ccc(C)cc2)CC1)OC)OC c1(OC)ccc(C(C(=O)N2CC(NC(C3CCCCC3C(N)=O)=O)C2)OC)cc1 C12(NC(=O)C=CBr)CCCC1CN(C(c1cccc(CN3CCCCC3)c1)=O)C2 C(C)(CCC(=O)NCCN(C)C(c1cc(OC)cnn1)=O)OC C1(C(N(CC(C)O)CC)=O)COC(CNC(c2ccc(C)o2)=O)C1 C1(NC(C2CC(C)(NC(=O)CCc3csnn3)C2)=O)CC2(CCC2)C1O O=C(C1=CCOC1)NCCCN(CCO)C(C1CCCOC1c1cc[nH]n1)=O c1(C(N(CCCN(C)C)CCNC(=O)CC2CCC(O)C2)=O)[nH]nc2ncccc12 C(C#CC(F)(F)F)NC(CCOCCCNC(Cc1c(C)ncs1)=O)=O N1(CCc2nccc(C)n2)CCC(=O)N(CCCN(c2ccccc2)C2CC2)C1=O C1(NC(CN(c2ncccn2)C)=O)CCCN(C(=O)CSC2CCOC2=O)CCC1 c1(-c2nc(CNC(C(C)(C)O)=O)sc2)ccc(F)c(Cl)c1 C1(C(=O)NCC(c2ccccc2F)NC(c2n(CC)ccn2)=O)(OC)CCCOC1 N1(C(C(=O)NCC)=O)CCC2CCC(C1)N2C(=O)Cn1nc(C)c(Cl)c1C Cc1c(CNc2cccc(C(=O)NC3(c4ccccc4Cl)CC3)c2)cccc1O N1(C(CNC(CC)=O)=O)CC2CC2C1C(=O)NCC1CCOC1 CN1CCCCC1C(N1CC(O)(CCNC(=O)C(C)(C)N(S(C)(=O)=O)C)C1)=O c1(C(N(CC(=O)NCC(CC)NC(=O)Cn2nccn2)C)=O)cc(C)nc(O)c1 C1(C(=O)NCc2c(C(N(CC(F)Cl)C)=O)con2)C2CC3C(C2=O)C13 c1(OC)cc(NC(C23CC2CN(C(C2(C)CCCN2)=O)C3)=O)cc(F)c1 Cc1nc(N)cnc1C(=O)N(C)CC1CCN(C(=O)C=CS(C)=O)C1 N1(C(Cc2ccc(C)o2)=O)CCCC(O)(CO)C1.N12CCC(C1)C2=O c1(C(C(=O)Nc2ccc(F)cc2)N(C(C2CCC2)C)C)ccc2c(c1)CCC2 c1(C(N(C2CCCN(C(=O)Cc3cnsc3)C2)CC)=O)cncc(OC)c1 CN1CCN(C(=O)C(C2CCCO2)CC(=O)O)CC1 c1(C(N2CCCCC(NC(c3cccnc3)=O)C2)=O)cc(Cl)c(Br)c(Cl)c1 c1(CC)noc(C(=O)NCC2(NC(=O)CS)CCOC2)c1C.n1(C2CC2)ccnn1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC2(CC2C(=O)NCCCCC2CC2)C1 c1(N(C)C)ncccc1C(=O)NC(C)(C)CCNC(C1CCC(C(N)=O)C1)=O CCC(CC)C(C(=O)NC12CC1CN(C(C1CCC13CCC3)=O)C2)OC c1(C(=O)NC(C2CN(C(C3(CO)CC3)=O)CCO2)C)cccnc1-n1cccn1 c1(NC(N2CCC2COC(Cc2c(C)noc2C)=O)=O)cncc(S(C)(=O)=O)c1 C(=O)(C1=NOC2COCC12)N(CC(C)C(=O)NCCC1CCCCO1)C C1(C(N(CCN(C)C)CC)=O)COC2(C1)CN(C(=O)C(C)(C)C(C)C)C2 N1(C(c2ccc(OC)nn2)=O)CCC2CCN(C(=O)CC3CS(=O)(=O)C3)CC12 c1(C(N(CCN(C(CC=CCC)=O)C(C)C)C)=O)cnn(C2CCC2)c1C c1(CC)ccc(OC)c(C(N2C3CC2CN(C(=O)COCC2CCCO2)C3)=O)c1 Cc1cc(Cl)nc(N)c1C(=O)NCC(O)CNC(=O)CCc1cncs1 c1(OC)cc(NC(C2CC(C)CN(C(=O)CCCC3CCCO3)C2)=O)cc(F)c1 CN1CCN(c2ncc(C(c3nnnn3C3COC3)NC3CSC3)s2)CC1 c1(C(=O)NCC2CC(OC)CN2C(C2COC2)=O)cn2cc(Cl)cc(Cl)c2n1 C1(C(=O)Nc2nc(Cl)ccc2C(F)(F)F)CCCC2(CCOC2)O1 c1(CC)noc(C)c1CNC(=O)N(C(C)Cc1ccccc1)CC CCC(C)C(C(=O)NC(Cc1ccco1)C(=O)NCC(CC)C(C)C)N(C)C N1(C(c2cc(CC)nn2C)=O)CCCC2(CCN(Cc3cc(C(C)C)no3)C2)C1 C1(CNC(C)=O)(NS(=O)(=O)CC)CCN(CC2(CC(=O)OCC)CCCC2)CC1 C(=O)(CC1OCc2ccccc21)NC(C)CNC(c1coc(CO)c1)=O c1(C(C)NC(C(C)NC(CCc2cc(C)no2)=O)=O)c(C)noc1C N1(C(C(=O)NCC(c2ccccc2)N2CCOCC2)=O)CCC12CCCOC2 C1(N(C(c2cn(CCC(C)C)nn2)=O)C)CCCN(c2cc(O)ncn2)C1 C1(NC(CC=C)=O)CN(C(c2ncc(Cl)s2)=O)CCC12CCCC2 N1(C(COC(C)C)=O)CC(CNC(c2nn(C)cc2Cl)=O)C2(CC2)C1 CC1(NC(=O)C(C2CCCC2)C2CC2)CCCCCC1 CC1CCCN(C(=O)C=CCC(C)(C)NC(=O)C(=O)NCCC(N)=O)C1 N1(C(CCCC#CC)=O)CCC2CN(C(=O)CCCCCc3cccs3)CC12 C1(CC)CN(C(=O)C=CC2CC2)CCN1C(c1cccc(I)c1C)=O C(=O)(C#CC1CCCCO1)N1CC2C(NC(c3sccc3C(F)F)=O)(CCC2)C1 c1(-c2n(C(CC)C)ncc2)cc(C(=O)NC2(N(C)C)CCCC2)c2cc[nH]c2c1 c1(C(N2CC(c3cn(CC=C)nn3)(F)C2)=O)cnn(Cc2ccc(F)cc2)c1N C(=O)(C1Cc2ccccc21)N1CC(C2(NC(c3scc(C(N)=O)c3)=O)CC2)C1 N1(C(=O)OC(C)(C)C)CC(O)CC1C(=O)NCCNC(C1CC1C1CC1)=O CC(Cc1ccncc1)C(=O)NCCC(O)CNC(c1sccc1C1CC1)=O Cc1cn(C)cc1Cc1cn(C2CCC(C(N3CCCCC3CO)=O)CC2)nn1 C1(NC(c2n(C)ncc2Cl)=O)CCCN(C(c2ccc(OCCF)cc2)=O)CC1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)N2)C)=O)ccc(O)nc1Cl C(=O)(C(C)(C)CCCNC(C1CCCSC1C)=O)N(CCN(CC)CC)C C1(CNC(C(N2CCNC2=O)C)=O)COCCN(C(=O)C(c2ccccc2)C)C1 Cc1ccc(F)c(CC(=O)NC(C)CC2CN(C(c3cc([N+](=O)[O-])sn3)=O)C2)c1 c1(C(=O)NCC23N(C(c4c(C)nccc4)=O)C(CC2)CC3)c(Cl)sc2nnsc12 C1(CC(=O)NCC(C2N(C(C=CC(C)C)=O)CCCC2)(C)C)CC2(CCC2)CCO1 n1(CC(N2C(CNC(C(CC)N(C)C)=O)CC2)=O)nc2n(c(=O)c1=O)CCC2 c1(C(N(C2CCN(C(c3cn(C(F)F)cn3)=O)C2)C)=O)ccc(O)cc1F C(C)(CS(N)(=O)=O)NC(=O)C=CC(=O)N(C1CC1)CC1(CCOC)CC1.C(=O)N C1(CNC(c2cc(C)[nH]n2)=O)CC(C)CN(C(=O)CN2CCOCC2)C1 C1(C)(C(=O)NC2C(C)CN(C(c3ncccc3C(F)F)=O)C2)CCCCCC1 CN1CCC(C(N2CCC(O)(CN(C(=O)C(CO)N(C)C)C)C2)=O)CC1=O c1(CC)nc(C(=O)NCC(C(C)C)NC(c2csc(CC(C)C)n2)=O)co1 C1(O)(CNC(C2(CCN(C)C)CCCC2)=O)CCN(C(=O)CCc2ccoc2)C1 c1(C(=O)NC2CN(C(C(C)CC3CCCC3)=O)CC2C)ccc(P(C)(C)=O)cc1 C12(C(=O)NC3CN(C(c4cnn(CC)c4Br)=O)C3)CCCCC1CCC2 c1(C(=O)NCCC(CNC(C=C(C)C(C)C)=O)O)ccccc1SC(F)F C1(CNC(CCNC(C)=O)=O)CN(C(=O)CC2CC=CC2)CCC1(C)C C1(O)(CCNC(c2cc(CNC(CC3C(C)CCO3)=O)sc2)=O)CCCCC1 CC1(CNC(=O)CC2CC(F)C2)CC(F)(F)CN1C(c1cc(O)cc(O)n1)=O C1(C#CC(=O)N2CCCC(CN(C(=O)C(F)(F)C(F)F)C)C2)(CC)CC1 N1(C(c2cccc(C)c2C)=O)CCCN(C(=O)CC(F)F)C(C)C1 C(C1c2ccsc2CCN1C(=O)CCCS(C)(=O)=O)NC(CCN(C)CC)=O C(=O)(C(CO)C(C)(C)C)NCC1CN(C(Cc2ccc(C)cc2)=O)C1 N1(C(=O)Cc2ccc(Cl)c(Cl)c2)CCOC2(CCN(C(C3(O)CCC3)=O)C2)C1 N1(C(c2cnn(C)c2F)=O)CCN(C(c2ccc(C(=O)O)[nH]2)=O)CC(CO)C1 C1(CC)(CNC(=O)C(CNC(=O)C=CCO)N(C)C)CCOC1 CC(C)(C)C(CNC(c1cccc(C2CC2)n1)=O)NC(c1cnc(C2CC2)s1)=O C=C1CC(C(=O)NC2(c3cccs3)CC2)(CNC(C2CCCN2C)=O)C1 C12(C(=O)NCC3(F)CCN(C(Cc4nnc(C)o4)=O)C3)CCCCCC1OCC2 O=C(N=c1ccn(C2CC2)[nH]1)C1CC2CC2N1Cc1cccc(F)n1 C(=O)(C1=CCCSC1)NC1C2CC(NC(C(CC)C#N)=O)CC21 c1(C(=O)NC(CNC(c2nn(CC)nc2C)=O)C2CC2)cccc(C(C)C)c1N Cc1cc(C(N2CC3CCC3(CCNC(c3cc(F)c[nH]3)=O)C2)=O)cc(O)n1 Cc1ccc(C(=O)NC2CC(NC(=O)C(C)(O)c3ccccn3)C2)cc1 n1(C(=O)NCC2N(CC(=O)NC3CC3)CCC2)nc(C2CC2)cc1C(F)F c1(NC(=O)NC2C3CCC2CN(C(C2(C4CC4)CC2)=O)C3)ccccc1[N+](=O)[O-] C1(C2CCN(C(c3ccc(Cl)c(C)c3)=O)C2)(NC(c2n(CC)cnn2)=O)CC1 C(CN=C(NCC1CCC(CC)O1)NC1CS(=O)(=O)c2ccccc21)OCC N1(C(C(CCC)O)=O)CC(F)(F)CC1CNC(C1CC(CF)C1)=O N1(C(CCC(C)c2ccccc2)=O)CCCN(CCNC(=O)COCCF)CC1 C1(C(=O)NCC(C)(C)C(=O)NCCCn2cnnn2)CCCC12CCC2 Cc1cc(CN2CC(C)(C(=O)Nc3cc(Br)ncc3C)C2)ccc1O CC(C)C(C)CC(=O)N1CCCC1Cc1ccccc1 c1(C(=O)NCCCN(C(=O)C=CC(C)C)CC)cc(N)cc(O)c1 Cc1nc(NC(C2CCN(C(C3CCSC3)=O)C2)C)cc(O)n1 N#Cc1cnc(NC(=O)NC2CCC(NC(=O)C3CC3)CC2)c(C#N)c1 c1(OC)nccc(C(=O)Nc2cc(-c3ccc(C)c(C)c3)[nH]n2)c1Br N(C1=NCC2CCCCN12)C(c1ccc(N2CCC(C(=O)N(C)C)C2=O)cc1)C N1(C(C2(CC=C)CC2)=O)CCC(NC(c2cc(COC)[nH]n2)=O)C1(C)C N1(C(C#CCNC(C2N(C)CCC2)=O)=O)CCC2CCCC2C1 C1(CNC(C2(CCC)CC(=O)C2)=O)CCCN(C(=O)C=Cc2cn[nH]c2)CC1 N1(C(C2(CC)CC(C)(C)C2)=O)CCC(C)C(C(=O)N(C)Cc2cncnc2)C1 c1(OC)ncnc(C)c1NC(c1csc(CNC(=O)CN2CC3CCC2C3)c1)=O C1(COCC(=O)NC2CC2)CN(C(c2cc(C(O)C(F)(F)F)ccn2)=O)CCO1 C(=O)(CCCCCF)N1CCC(C(CNC(C(CC)C)=O)O)CC1 C12(NC(CC3(N(C(CCC(C)CN(C)C)=O)C)CC3)=O)CC1COC21CCC1 CC1CC(NC(c2cc(C3CCC3)on2)=O)CCN1C(c1nc(Cl)sc1Cl)=O CS(=O)(=O)CCCC(=O)N1CCCC(CO)(NC(=O)CCN2CCCC2)C1 c1(OCC)cc(C)ccc1NC(c1cnccc1Nc1ncc(CO)[nH]1)=O c1(C(=O)NCC2CCC(NC(C3CCCCC3O)=O)CC2)ccc2c(c1)OCC2 C(=O)(C(Cn1cncn1)NC(=O)C=Cc1ccco1)N(C1CCC1O)C C1(NC(c2csc(C)c2N)=O)CC2CC1CN(C(=O)C1=C(Cl)CCOC1)C2 C1(C(=O)NC(c2cccs2)COC)CCCN(c2cc(O)nc(C)n2)CC1 c1(C(N2CC(OC)(CNC(C3COC(C)C3)=O)C2)=O)cnc(N)c(N)c1 CC1CN(C(c2cccnc2O)=O)CC(C)C1NC(c1ccc2occc2n1)=O CC1(C)C(C(=O)NC(C2CCCCC2)CO)CCN1C(C1CC(n2cccn2)C1)=O N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(c2cccc(F)c2Cl)=O)CCC1C Cc1cc(CCC(=O)NCC2CC2NC(c2c[nH]cc2C)=O)c(C)s1 N1(C(c2c(CNC(c3nc(C)sc3)=O)ccs2)=O)CCC(=O)N(C)CC1 N1(CCC(=O)NCC(C)CNC(c2c[nH]c(C(N)=O)c2)=O)CCP(C)(=O)CC1 c1(CC(=O)NCCNC(C2CC(N(C)C)CC2O)=O)cccc(O)c1F C1(NC(CCCCCC)=O)CC2CC1CN(C(=O)CC1OCCCC1(C)C)C2 C1(CCNC(C2CN(C)C2)=O)CCCCN1C(=O)Cn1cc(CO)nn1 C12(NC(C3(C(F)(F)F)CC=CC3)=O)CCN(C(=O)CCF)CC1C2 n1(CC)ncc(C(=O)NC2COCCC2NC(c2ccccc2C)=O)c1C C1(NC(COCCOC)=O)C2CCC1CN(C(=O)CC1CC3(CC3)CO1)C2 N1(C(C(C=CCCC)O)=O)CCCC(C2CN(C(C3CC(C4CC4)=NO3)=O)C2)C1 c1(C(=O)NCC2C(C(=O)NCCN=[N+]=[N-])C2)cnc(C2CC2)[nH]1 C1(C(=O)NCc2occ(C)c2)CCC(O)CN1C(c1cccnc1C)=O CC1(C(N2CCC(C(=O)NCCCSCCO)C2)=O)CC2CC2C1 C(CC(CC)C(=O)NCCCCN(CCCNC(c1cc(F)cc(F)c1)=O)C)=CC C1(NC(CCC)=O)CC12CCN(C(=O)Cc1ccc(OCC)nc1)CC2 c1(OC)ccc(C(N2CCC(c3cncn3C)CC2)C(=O)NCC(F)F)cc1 Cc1cc(Cl)ccc1OCC(N1CCC(NC(=O)C2=CCC2)C(C(C)C)C1)=O CC(F)(F)CCC(=O)NCc1ccc(C(=O)NCc2nccn2C2CC2)o1 C=CCN=c1[nH]c(C(N2CC3(CNC(c4cnc(CC)s4)=O)CC2CO3)=O)cs1 c1(CN(C(=O)CCC2CCCN2C(c2ccoc2Cl)=O)C)cccc(F)c1 Cc1cnc(CNC(C2CC23CCN(C(=O)Cn2[nH]cnc2=N)C3)=O)c(C)c1 c1(OC)ccc(OC)c(C2CN(C(=O)CCCCNC(N)=O)CCN2CC#N)c1 N1(C(C2C(C)C2C)=O)CCC2(CC1)CN(C(c1ncccc1Cl)=O)C2 c1(C(N2CC(CC(N3CCC(=C)C3)=O)OCC2)=O)cccc(OC(F)F)c1 C1(C(N(C)CCC2CCNCC2)=O)C2CN(S(=O)(=O)CC3CCS(=O)(=O)C3)CC12 C12(OC)CCC(C(=O)NC(C)(C)C(C)NC(c3ccc(Cl)cc3C)=O)(CC1)C2 c1(C(=O)NCC2CCC(NC(c3nc(CC)sc3)=O)C2)ccn2ccccc12 C(=O)(CC(C)CCC=C(C)C)N(CCC)CCNC(C1CCC2CC12)=O CC1CC(F)(F)CCN1C(C1(CCNC(=O)COCC2CCCC2)CCCC1)=O N1(C(c2cc(C)[nH]n2)=O)CC2CC1(c1cn(CC(=O)O)nn1)CO2.N12CCC1C2 c1(NC(C2OCCC(NC(C(C)(O)CCl)=O)C2)=O)cccc(F)c1F c1(-n2cc(C(C)NC3C=CCCC3)nn2)cccc(S(C)(=O)=O)c1 C1(N(C)CC)CCN(C(=O)CCC2CCN(C(=O)C(C)n3ccnn3)C2)C1 C1(C(N(CC#C)CC2CCC2)=O)CC(NC(=O)CC2CNC(=O)O2)CCO1 c1(SOC(C)(C)C)ncccc1F.C12CCCN1C(=O)C1(CCC1)CN(C)C2=O C1(CNC(CC2(OC)CN(C(c3cc(=O)n(C)cn3)=O)C2)=O)CCC(=O)NC1C O=C(C1=NOCC1)NC1CCCC(NC(c2cc(C(F)(F)F)ns2)=O)C1 C1(C)(CNC(CC2N(C)CCCC2)=O)COCCN(C(=O)CC2CC3(CC3)C2)C1 C(=O)(CC(C)(C)C(F)F)NCCC(CNC(c1ncc(C)cc1F)=O)O C1(CC(=O)N(CCC(=O)NCCCN(C)C)CC=C)C=NN(C)C1=O N1(C(c2nccc(C(=O)OCC)c2)=O)CC(C)CN(C(C2C=CCS2)=O)CC1C Cc1ccc(C=CCNC(C2CCC(n3cc(C4(O)CCC4)nn3)C2)=O)s1 Cc1ccccc1N=c1[nH]nc(CNC(=O)CC2CN(C3CCOCC3)C2)s1 C1(NC(CN(C2CCSC2)C)=O)C=CCN(C(C2CCS(=O)CC2)=O)C1 C1(NC(c2cc(C(F)(F)F)cc(C(F)(F)F)c2)=O)CCCCCCC1(F)F C(=O)(C(C)(O)C(C)(C)C)N1CCC(n2cc(CC(COC)O)nn2)CC1 O=C(C1=NOC2(CCC2)C1)NCCC1CN(C(=O)C=CCn2cncn2)CCO1 C1(NC(C(CC2CCC2)NC(c2n(C)ccc2)=O)=O)CCN(C2CC2)CC1 c1(CC)cc(=O)oc2cc(OOC(=O)C(C)Cc3cnn(C)c3)ccc12 N1(C(CC2(C)CCCO2)=O)C2CCC1C1CC1(NC(=O)CCc1cc(Cl)no1)C2 c1(OC)cc(C(=O)NC23CC(NC(C4CCC(=O)O4)=O)(C2)C3)cnc1O CN1CCC(C(N2CC(C(N)=O)(CNC(c3ocnc3C(F)(F)F)=O)C2)=O)C1=O Cn1ccc2cc(C(N3CC4CC(C3)N4C(=O)C(C)(C)CCl)=O)ccc12 c1(C(=O)NC(CNC(C(COC)N(C)C)=O)C)cc(Cl)nnc1O N1(C(C(C=C)(C)O)=O)CC2CCCC(NC(=O)CN3Cc4ccccc4C3)C2C1 C1(NC(c2ncc(C)c(C)c2)=O)CN(C(=O)C=CC(C)C)C2(CCCC2)C1 C1(C(=O)NCC(C)CC(=O)NCC2CC2(C)C)CC2(CCO1)CC2 C(C1=CCCOC1)NC(=O)CCC1(N(C(C2CC2c2ccoc2)=O)C2CC2)CCC1 c1(C2C(C(N(CCOCCN(C(CC(=O)OC)=O)C)C)=O)C2)ccnc(C)c1 S(=O)(=O)(c1cnn2ccc(N3CCc4oc(C)nc4C3)nc12)N(CC(CC)C)C c1(C(C)=O)c(C)[nH]c(C(N2CCCC(C(C)NC(c3coc(Cl)c3)=O)C2)=O)c1C C(=O)C1=COCCC1.n1(C(=O)OC)nccc1C(=O)OCCN(C(C)=O)C N1(C(C2(C)CCC(=O)N2)=O)CCC2CN(C(C3CN4CCN3CC4)=O)CC2C1 c1(C(=O)NCC2(C(C)(C)O)CN(C(CCC=CC)=O)C2)nc(SC)ncc1Cl C1(C(=O)NCC2CCN(C(CC)=O)CC2)CCc2ncc(Br)n2C1 CC1=NOC(C(=O)N(C2CCN(C(=O)Cc3csc(-c4ccco4)n3)C2)C)C1C C(C(C)(O)C(C)(C)C)NC(CCC1CC(NC(C(C)N=[N+]=[N-])=O)C1)=O C(C)(CNC(=O)C(CO)NC(N)=O)(C(C)C)NC(Cc1cc(C)on1)=O O=C1COC(C(=O)NCC2CN(C(=O)Cn3ccsc3=N)C2)C1 C(=O)(C(CC(C)C)C1CCCCC1)N(CCCCNC(C=CCC)=O)CC N1(C(c2c(Br)ccc(CC)c2)C(=O)O)CCCC(C2CN(C(C)C)C2)C1 C(C1CCCN1C(=O)CC(Cl)Cl)=CC(=O)NC1CCCC1F C(CN1C(=O)NCC2CC(OC(c3ccc(C)cc3C)=O)C2(C)C1)OC Cc1ccc(NC(C2(CNC(c3cc4n(n3)CCC4)=O)CCCC2)=O)cc1F N#CC1CC2(CN3CCCC(OCc4ccccc4)C3)CC1C2 N1(C(C(C=C)CC)=O)CC(C)CN(C(=O)CCCc2cnn[nH]2)CC1C N1(C(C2(C3CCC3)CC2(F)F)=O)CCC(F)(F)C(CON)C1 C(=O)(C(CC)C(C)C)N(CCNC(CCOCC#C)=O)C C=Cc1cnn(C)c1C(=O)NCCCCC(C)NC(=O)CCCOCCC c1(C(=O)NC2CN(C(c3cnc(OC)s3)=O)CC2C(F)(F)F)ccc(F)c(N)c1 c1(C(N2CCN(CCOC)CC2)C(=O)NCc2nnn(C)n2)cc(C)cc(C)c1 C1(CNC(C2C(CC(C)C)C2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CC(NC(CNC(c2cc(C)sn2)=O)=O)C1 C(=O)(C(CC(C)C)NC(C1C=CCN(C(c2ncc(Cl)cc2Cl)=O)C1)=O)NC N1(C(c2nc(CC)oc2C)=O)CCCN(CCNC(=O)Cc2csnn2)CC1 c1(NC(CC(=O)NC)C)[nH]c(=NC2COC3(CCCC3)C2)nc2sccc12 C1(C=O)CC(=O)N(CC(N2CC(CCC34C5CC3C3C4C53)C2)=O)C1.CC=O C12(COc3c(C)nns3)COC(C(=O)NC3CCN(C(c4cn[nH]c4)=O)C3)(C1)C2 Cc1nccn1CC(N1CC(C(C(=O)NCCCC(F)F)N(C)C)C1)=O C1(NC(=O)CC=C(Cl)Cl)CC(NC(c2ccc(Br)cc2)=O)C12CCC2 C=CC1CN(C(=O)C(C)N(C(=O)CCNC(C)=O)C)C1 C1(NC(=O)CCc2ccsc2)CCC2(CC1)CC(NC(=O)C(F)CC1CCC1)C2 c1(C(=O)NCC2(CCNC(CCC(CC)C)=O)CC2)cc2c(F)cc(F)cc2o1 N1(C(C2CCC(C(C)C)NC2=O)=O)CCC2(CC1)CN(C(=O)Cn1cnnn1)C2 C12(C(N(C3CCN(C(C(C=CCCC)O)=O)CC3)C)=O)CCC(CO)(CC1)CC2 C12(C(=O)OCC(c3ccc(OC)nc3)=O)CC=CCN1CCC2 c1(C(N2CC(N(C(C(C)CC(N)=O)=O)C)C2)=O)cc(C(F)(F)F)ncc1[N+](=O)[O-] c1(C(N2CCC(C(C(=O)NC(CCCC=C)C)(C)C)C2)=O)c(C)cccc1F c1(N2CCC(CNC(C3(C)CCC(C)C3)=O)C2)ncccc1C#N C1(NC(c2n(CC)ncc2)=O)CCCC12CN(C(=O)CC1(CO)CCCC1)C2 c1(C(N(CC(C)NC(C(CC)OCC)=O)C)=O)cnc2ccncc2c1 C=C1CCC(C(N2CC(NC(c3ccc(CSC)o3)=O)C(O)C2)CC(C)C)CC1 c1(C(=O)NCC(CC)NC(c2csnc2Cl)=O)ccc(Cl)c(C(C)=O)c1 N1(C(c2ccc(-c3ccc(=N)[nH]c3)o2)=O)CCCCC(CNC(=O)C=C(Cl)Cl)C1 CCC1=NOC(C(=O)N(C)CC2CCN(C(=O)C(c3ccc(Cl)cc3)=O)C2)C1 C1(C(=O)NCCC2CCCC3CC23)CC2(CCC2)CN1C(=O)C(O)C(F)(F)F c1(C(N2C3C(NC(C4(COCC)CC4)=O)CC(C3)C2)=O)nccc2occc12 c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(NS(=O)(=O)CCc3ccccc3)C2)n1C N1(C(c2cc(C)[nH]c2)=O)CCC2(NC(=O)CC3CCNC(=O)C3)CCCCCC12 C1(CNC(C2(OC)CCCOC2)=O)CN(C(C2CSCC(=O)N2)=O)CCC1C C1(F)(CNC(C=CC(C)(C)SC)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1 CC(CCCC(=O)N1CCOC(CCCNC(=O)CCn2cccc2)C1)N(C)C O(N1CCC(CC(=O)N(CCCOCC)C)CC1)CC.C(=O)(CCC1CCCO1)NC C=CCC(Cc1ccccc1)C(=O)NCC(C1CC1)NC(C1(CO)CCCC1)=O Cc1cc(NC2CC(F)(F)C2)ncc1S(=O)(=O)NC1CC(COCC2CC2)C1 CN1CCC(CO)(CNC(=O)C(C)(CO)NC(=O)CN2CCNC(=O)C2)C1 C1(O)(CNC)CCN(C(=O)CCC(N)c2ccccc2)CC1 c1(OC)ccccc1CC(=O)NCC1C(C)CCN1C(=O)C=CCN1CCOCC1 C1(O)(CNC(=O)COCC2CC2)CCN(C(=O)CN2C(=O)CCC2=O)CC1 c1(OC)cc(C)c2cc(C(=O)NCC(C)CNC(c3ccc(F)cn3)=O)[nH]c2c1 C(C(CC(F)(F)F)NC(=O)C(C)SCC(C)C)NC(C1(OCC)CC1)=O N1(CC2CCC(C)CC2)CCCN(C(C2(C)CCOC2=O)c2ocnc2)CC1 C(C)(C(C)S(C)(=O)=O)NCC(CC(=O)OCC)c1ccccc1F c1(C(=O)NCC2(NC(C3C(SC)CCC3)=O)CCC2)ncccc1N c1(OC)ccc(-c2cncnc2NCc2cccc(C)c2Br)c(F)c1 c1(N2CCC(OC)(CNC(C3CC(C)CO3)=O)C2)cc2nnc(C(C)C)n2cn1 CCCCC(C)CCC(=O)NC1CC(OCC(=O)Nc2cnn3ccsc23)C1 N1(CCNC(c2cnc(Cl)[nH]2)=O)CCN(C(C2CCOC2C2CCC2)=O)CC1 c1(C(=O)NCC(C(C)C)NC(=O)C#CC(C)C)cc(S(N)(=O)=O)ccc1O CCCC(C(O)C(=O)N1C2CCC1CN(C)C2)NC(c1ccc(C)nc1)=O N1(C(c2nc(C(C)C)oc2)=O)CCCN(C(=O)CCOC2CCOCC2)C(C)C1 CC1CCCCC1C(N1CCN(CCCCCNC(=O)C=CC(F)(F)F)CC1)=O C(=O)(C1=CCCCC1)NC1CC(C)(NC(CC2(C)CC2)=O)C1 C(=O)(C1=C(C)CCCC1)N1CCCC(CN(C(c2ccc(OC)cc2C)=O)C)C1 N1(C(c2c(C)ocn2)=O)CC(F)CC1C(=O)NCCCc1cccnc1 c1(Cc2n(CCC#C)c(N3CCCC(CC)C3)nn2)cccc(F)c1F CC(CC(C)NC(=O)C=Cc1cn[nH]c1)NC(=O)C(C)(C)Nc1ccccc1 c1(C(N2CC(CNC(CCNC(=O)NC)=O)C(C)C2)=O)ccc2c(c1)CCO2 CC1CCN(C(=O)COc2cccnc2)CC1NC(c1cnnc(O)c1)=O c1(C(=O)NC2CCCC(NC(CCCC=C)=O)CC2)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)NC2CC(F)(F)CC2O)cc2cc(F)c(F)cc2[nH]1 C(=O)(C(CNC(=O)CCC(C)OCC)C(C)C)N(CCCN(C)C)CCC N1(C(CC(=C=C)C)=O)CC2(CNC(C3(C4CCCCO4)CC3)=O)CC1CO2 CC1=C(C(=O)NCC2CCN2C(C2CCCC(F)(F)CC2)=O)S(=O)(=O)CCO1 CC(C(C)(C)C(=O)N=c1cc(C2CC2)n(C)[nH]1)NC(c1ccoc1)=O CC(C)C(F)(CNC(c1cc(F)cc(F)c1)=O)C(=O)NCc1cc(C2CC2)n[nH]1 c1(C(=O)NC(CCC)CCCNC(=O)C(F)n2cccn2)cc(F)c(F)cc1O c1(C(N(C2CN(C(c3n[nH]c(C)c3O)=O)CC2F)C)=O)cc2n(n1)CCN(C)C2 C(C)(C(C(C)C)NC(=O)C=CC1CCCCC1)NC(COc1cc(C)on1)=O c1(C(=O)NC(CNC(C=CCC)=O)(CC)CC)ccc(OC)c(N)n1.NCC C(CCN=c1[nH]nco1)OC(c1cccc(OCC(C)C)n1)=O Cc1cn(C)cc1C(=O)NC(C)(C)CNC(=O)C(c1ccc(CC(C)C)cc1)C C1(C)(C(=O)NCCOCCN(C(=O)C(F)CC2CC2)C)CC1(F)Cl Cc1noc(Cl)c1CC(=O)NC(C)C(C(C)C)NC(c1ccsc1C#N)=O Cc1ccc(CC(=O)NC(C)CCNC(=O)C(C)NS(C)(=O)=O)cc1Cl c1(C(C(=O)NCC=C)N(CC(c2cccc(C)c2)(C)C)C)ccc(OC)cc1 c1(C(N2CCC(O)(CNC(C3CC34CC4)=O)C2)=O)cc2c(s1)CCCCCC2 S(=O)(=O)(c1ccc(OC(F)F)cc1)NCC1NC(=O)CC(C)C1.C1(C=O)CCOCC1 C12(CNC(C3(N(C)C)CCC3)=O)CC(CN1c1ncnc(Br)c1Br)C2 N1(C(C2CC(=O)OC2)=O)CCCC(n2cc(COCCCO)nn2)CC1 c1(SCC(=O)NCCN(C(=O)CSc2nnc(C)s2)CC)cccc[n+]1[O-] C(C)(CO)(C(=O)NCc1cc[nH]c1C(=O)N(C)C(c1ccncc1)C)OC C1(N(CC(=O)N(CC(C)O)CCO)C(=O)CC2CCCCC2)(CCO)CC=CC1 c1(C(=O)NC2CC3CN(C(c4nc(OC)oc4)=O)C2C3)ccc2c(c1)COC2 CC(C)CCC(O)C(=O)NCC(CNC(c1ccc(C(=O)N(C)C)cc1)=O)CO c1(C(N2CC(C(C)NCC3(C)CCCC3)C2)=O)cc(N2CCCC2)ncn1 c1(C(N2CCC(CC(=O)Nc3c(OC)cccc3)C2)=O)cc2cc(Br)ccn2n1 C1(C(=O)NCC=CCOC)C2CC3C(C2NC(C2CC2C(N)=O)=O)C13 c1(SC)cccc(C(=O)NCC(C)N(C)C(C2CCC(C(C)(C)O)CC2)=O)c1 c1(CC)ccccc1CC(=O)N(C1CCCCC1NC(C1(C)CC1)=O)C c1(C(N2CCN(C(C(C=CC)O)=O)CC2C(F)F)=O)coc(S(=O)(=O)NC)c1 c1(OC)ccc(S(=O)(=O)N2CCOC(CNC(C3C4COCC34)=O)C2)cc1 Cc1ccc(F)c(C(=O)NC2C3CC2N(C(c2nc(C4CC4)oc2C)=O)C3C)n1 Cc1cc(C(N2CCN(C(c3ccnnc3C)=O)CC2C)=O)c(C)n1C C12(NC(=O)Cc3cc[nH]n3)COC(C1)C(NC(c1cnc(-c3ccoc3)s1)=O)C2 S(=O)(=O)(c1ccc(F)c(F)c1)N1CC(C(=O)Nc2ncc(Br)nn2)C(F)(F)CC1 c1(NC(=O)C(c2cc3cnccc3o2)N2CCC(F)(F)C2)cccc([N+](=O)[O-])c1 N1(C(C(C=C)C)=O)CC2(CCCC2CC(N2CCn3nccc3C2)=O)C1 C1(C(=O)NCC(C)O)CN(C(c2ccn(C(F)F)n2)=O)CC12CC2 Cc1cc(Br)c(F)cc1NC(=O)C(=O)NC(CO)C(O)c1cccnc1 C1(OC)CC(F)CN(c2nnc(-c3ccc(Br)s3)n2CCC(=O)N(C)C)C1 n1(CC=CC2CCCN2C)cc(CCNC(=O)OC)cn1 c1(OC(C)C)ccc(Cl)cc1C(=O)NCC(C)(O)CNC(=O)CCCCC#N C1(O)(CNC(C2(C(C)C)CC2)=O)CCCN(C(=O)CCc2cnco2)CC1 N1(C(CCCC#C)=O)CC(C)CN(C(=O)CCNC(=O)OC)CC1C Cc1cc(C)n(CC(N2CC3CCC3(CNC(=O)C(C)(C)N(C)C)C2)=O)c(=O)n1 C(=O)(C1CCCc2cncn21)N1CC2(CCN(C(CC(C=C)CC)=O)C2)C1 S(=O)(=O)(c1ccc(C#N)c(N(C)CC2CCSC2)c1)N1CCCC(C=C)C1 CC(CN=c1nc2scnc2c(NCC(C)(F)F)[nH]1)C(C)(F)F N1(C(C2(c3ccccc3)CCN(C)C2)=O)CCN(C(=O)CC2CC2)C(CO)C1 Cc1ccnc(C(=O)NC2(CNC(=O)CC(C)(C)C3CC3)CCCC2)c1F C(=O)(CCC1=NNC(=O)CC1)N(C1(C)CCCCN1C(=O)OC(C)(C)C)C(C)C CC(C)(C)C(=O)C(=O)NC1CN(C(c2c(O)cccc2F)=O)CCC1C(F)(F)F CN1CC(C(=O)NC2CC(CCOCCNC(=O)COC3CCOC3)C2)NC1=O c1(-c2nc(NC(C(Cc3cccc(OC)c3)N)=O)sc2)cc(F)ccc1F C1(O)(CNC(=O)C(O)C2CCC2)CCN(C(C2CC2(Br)Br)=O)CC1 Nc1ccc(NC(=O)NC2(c3ccc(F)cc3F)CCC2)cc1Cl C1(CNC(c2nccc(C)c2F)=O)CN(C(C2CCC3CC2C3O)=O)CCCO1 C1(NC(=O)C=C2CCC2)CCCN(C(c2ccncc2)=O)CC1F C1(CN(C)C(C2(C)CC2Br)=O)CCCN1C(=O)CN1CC(F)(F)C1 C1(C(=O)NC2CCN(C)C(=O)C2)C(C2CC2)CCN1C(=O)CCC(N)=O C12CCC1(CC)CNCCNC2=O.c1(SCC)cnc[nH]1.C(CC)N(CC)CC Cc1sc(N)c(C(=O)NC2CCC2NC(=O)C=Cc2cccs2)c1C c1(CCC(N2CCC(O)(CNC(C(CC#C)C)=O)C2)=O)ccc([N+](=O)[O-])cc1 N1(CC(=O)N(CC(N)=O)C)CCC(N2CC=CC2)C1 c1(OC)ccc2ccccc2c1CNc1ccc(C(=O)OC(=O)C(F)(F)F)cc1 c1(C(NNC(C2N(c3ccc(C)nn3)CCC(=O)N2)=O)=O)cccc(S(C)(=O)=O)c1 C1(CN(C(=O)C(CO)c2ccccc2)C)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 C(=O)(CCCC(F)F)NC1C(OC)CN(C(C2CC(F)(F)C2)=O)C1 C1(C(=O)NCC(CC)(CC)OC)Cc2ccccc2CN1C(=O)CSC1CC1 N1(C(CN(C(C(C)OCC=C)=O)C2CC2)=O)CC=CC1CSC C(=O)(C1=NNC(=O)CC1)NC(C1CCCN1C(C1OCC1(C)C)=O)C c1(OC)ccc(C(=O)NCC(C2CC2)N(C(=O)C(C)n2ccnn2)C)c(O)c1 c1(C(=O)NCC(CC)NC(=O)CCCC2CC2)nc(Cl)nc(SC)c1C C(=O)(CCC(F)(F)CN=[N+]=[N-])N(C1CCN(C(CC(COCC)C)=O)CC1)CC C12(C(N3C4C(CNC(c5c(C(C)C)ccs5)=O)C(C4)C3)=O)CCCC1CC(=O)C2 CC(CCCNC(=O)CC1(O)CCCC1)NC(C1(c2ccno2)CCC1)=O CCCC(CCCO)C(=O)NCC1CCCCC1NC(c1csc(C2CC2)n1)=O C1(c2nnnn2C)(NC(C23COC(CF)(C2)C3)C)CC2CCOC12 CCCS(=O)(=O)C(C)C(=O)NCC1CC2(CC2)CN1C(=O)CNC(=O)CN(C)C C12(CC(=O)NC(CC=C3CC3)=O)CCC1CN(C(c1nonc1N)=O)C2 CC1(C)CC(NC(C2(C)CCCN(C(C3(CCN=[N+]=[N-])CC3)=O)C2)=O)CCO1 N1(C(c2c(CNC(C(C)OC3CCCC3)=O)cco2)=O)CCS(=O)C(C)C1 CC#Cc1cncc(-c2cscc2C(=O)NC2(C#N)CCOCC2)c1 C#CC1CN(C(=O)CC2CCCCC2)CCN1C(c1cc2nccnc2[nH]1)=O C(=O)(C1=NOC(C)C1)NCC1CCCC1NC(N)=O.Cc1nc2oc1C(=O)NC2 c1(C(N2C(C(C)NC(=O)Cn3cc(Cl)cn3)CCCC2)=O)c[nH]nc1S(N)(=O)=O N1(C(C(CC)(C)C#N)=O)CCC2(CC1)CC(C)N(C(=O)C1=CS(=O)CCC1)C2 c1(CCC)cccc(CNC(=O)NC(Cc2cccc(Cl)c2)CO)c1 C1(CC)(CC)CN(c2cc(N3CCCC(c4ncc(C)s4)C3)ncn2)CCS1=O c1(C(N2C(C)CCN(C(C(CC)O)=O)CC2)=O)nccc2ccn(C)c12 c1(C(=O)NC2CCC(NC(c3n(CC)nc(C)c3)=O)C2)cc(C)ccc1C(F)F c1(C(=O)NCCN(C(C2C=CCCC2)=O)CC2CC2)ccc2nn[nH]c2c1 N1(Cc2c(CN(C)C)cccc2)CCCC(C)(C(=O)NCC2CC(=O)N2)C1 N#Cc1ccsc1C(=O)NCC1CCCCN1C(=O)CC1CC1(Cl)Cl N1(C(C(C(C)C)C2CCC2)=O)CC2(CCCC(CNC(C3(F)CC3C)=O)O2)C1 c1(N2CCC(CCOC)(NC(c3ccnc(C)n3)=O)CC2)ncc(C#N)cc1F Cn1ccc2cc(Nc3nc(C)cc(=NCC4CCCCC4(C)C)[nH]3)ccc12 N1(C(CC(=O)NCC)=O)CC2C(CNC(c3cccnc3CO)=O)C2C1 n12cc(nn1)CNCCC2.c1(C(=O)OC)coc(C2(C(F)(F)F)N=N2)c1 c1(OC)ccc(F)cc1NC(C1(O)CCN(S(=O)(=O)CCCl)CC1)=O.C12CC1N2 N1(C(CC(C(F)F)NC(C2(CCC)CC2)=O)=O)CCOCC(C)(F)C1 c1(C(=O)NC2CC(NC(c3cc(Cl)c(Br)[nH]3)=O)C2)cccc2c1CCOC2 CC(C)(Cn1nnnc1N1CCC(CC(N)=O)C1)CC(F)F c1(C(=O)NCC2(F)CC(NC(CC3C(CC)C3)=O)C2)cc2cc(C)ccc2o1 CCC(C)(COC)CNC(C1CN(C(=O)C(C(C)C)OC)CC1C)=O CC1(Br)CC1C(=O)NCCCN(C(=O)CSc1cccs1)C1CC1 C(=O)(CCCC(F)F)N1C(C2(NC(=O)CCc3cnccn3)CC2)CCC1 C(=O)(CC1OCCc2sccc21)NCCC1CN(C(Cc2c(C)cccc2)=O)C1 c1(C(=O)NC2(CF)CCN(C(C(CCSC)N(C)C)=O)C2)cc(F)c(C)cc1F c1(C(=O)OC)cnc(C)nc1NC1CCCN(C(=O)CCc2cncc(F)c2)C1 C1(C(=O)NCC(CC)NC(=O)CC2CN3CCC2CC3)CC1C1CCCC1 c1(C(=O)NC2C(C)CN(C(=O)CCC3CCCCC3)CC2)ncc2n1CCCC2 C1(NC(C(C)Oc2ccccn2)=O)CC2CCC(C1C)N2C(C1SCCS1)=O C1(C)(CCNC(CC2C(C)(C)CC2)=O)CCN(C(c2c[nH]nc2Cl)=O)C1 C(CS(=O)(=O)CC(=O)NC(C(N1CCC(OCCO)C1)=O)C1CC1)OC c1(C(=O)NC2CC(C)(NC(C=C(CC)CC)=O)C2)ccc2snnc2c1 c1(OC)nn(C)cc1C(=O)NC(C(=O)N1CCCC(CCOC)C1)C(C)O c1(NC(C)=O)nnc2cnccn12.c12ccccc1NC(=O)COC2=O CCCCCCCC(=O)N1CCCC(C2CCCCN2C(=O)CSC(F)F)C1 C1(C(=O)NC2C(NC(c3ccc(O)c(Br)c3)=O)C2)CC2(CCCC2)C1 C(CCC(=O)N1CC(O)(CN(C)C(C2CCC(C(N)=O)C2)=O)C1)OCCOC C12(F)CCCN(C1)C2c1cn(CC(n2cccn2)C)nn1.N1(CCO)CCOCC1 C(N=c1[nH]c(-c2ccccc2)nc(=NCCS(=O)(=O)CC)[nH]1)C1(C)ON=C(C)C1 N1(C(C2N(C(C)C)CCCC2)=O)CC(CO)C2(C1)CN(C(C1(N(C)C)CC1)=O)C2 c1(C(=O)NCC2(OC)CCN(C(C3CCCN(C)C3)=O)C2)cc(C)c(C)c(F)c1 c1(C(=O)NCC(C)N(C(C2CC2(C)C)=O)CC)ccc2cccc(OC)c2n1 C1(NC(CCN(C)CC)=O)CC2(C1)CC2NC(C1C(C#N)C1(C)C)=O c1(OC)ccc2c(n1)NC(C(=O)NC1CCCCN(C(C3CC=CCC3)=O)C1)C2 C1(C(=O)NC(c2nc(C)[nH]n2)C)CCN(C(c2ccc(CC#N)cc2)=O)C12CC2 C1(C(=O)NC(COC)CNC(c2n[nH]cc2Cl)=O)CCC(OC(F)F)CC1 N1(C(C(C)NC=O)=O)CCC(C2CC2)(CNC(=O)C=Cc2cccs2)C1 n1(NC(CCOC)(C)c2nnnn2C(C)C)cc(C)ccc1=O CC1C(NC(=O)C=Cc2ccccc2)CC2CCC1N2C(=O)C#CC1CC1 C1(C)(NC(C23CC(CN(C(c4c(C)ccc(O)c4)=O)C2)C3)=O)CC(C)(C)OC1=O C1(C(=O)NCC2(C(C)NC(C3CCOC3C(N)=O)=O)CC2)(N(C)C)CCCOC1 Nc1c(Cl)cc(C(=O)NC23CCN(C(=O)C=C4CC4)CC2C3)cc1[N+](=O)[O-] Cc1cc(C(=O)NC2CCCC(C(N3CCCC(OC4CC4)C3)=O)C2)cn1C c1(CC(Cn2cc(CC(C(=O)N(C)CC)C3CC3)nn2)O)ccccc1O c1(C(=O)NC2CC3CC(OCC)C3C2)c(C(F)(F)F)cc(F)cc1F C1(C)(CC(=O)N(C)CCOC)CCCO1.C1(=O)CN(C(=O)OC(C)(C)C)CCN1 Cc1ccc(C(=O)NC2(CCNC(=O)C(C)NC(C3CC3C)=O)CCC2)c(F)c1 n1(CC(N2CCC(CNC(C3N(C)CCC3)=O)C2)=O)ccc2ccccc12 c1(C(=O)NCC(CN(C)Cc2cc(O)nc(C3CC3)n2)O)cnc2ncccn12 N1(C(c2scc(CNC(CNC(N)=O)=O)c2)=O)CCC2(CCOCC2)C1 C1(CNC(CNC(C)=O)=O)CCCN(C(c2cccc(C3CNC(=O)C3)c2)=O)C1 C12(NC(C3CCC(C)CC3)=O)CCC(C(N3CCC(C(=O)N(C)C)C3)=O)(CC1)C2 c1(CC)cc(C(=O)NC2CC(NC(=O)CCNC(=O)OC)C2)cc(CC)c1 N1(Cc2occ(C(N)=O)n2)CCC(C(F)F)CC1 C1(COC)(CNC(C2CC(SC)C2)=O)CCN(C(=O)Cc2ncsc2Cl)C1 CC1(C)CCN(C(=O)C=C(C2CC2)C2CC2)CC1C(N1CC(c2nn[nH]n2)C1)=O C(CCO)(C(=O)NC(C)C(C)F)NC(C(N1CCCCC1)C)=O.C(CF)N C(C(CNC(c1ccc(CO)s1)=O)S(C)(=O)=O)NC(Cc1c(C)cccc1)=O c1(C(C)OCC)nc(CONC(c2ncoc2-c2ccco2)=O)cs1 N1(CC2OCC(C)(C)C2)CCCC(F)(CNC(=O)Cc2nnn(C(C)(C)C)n2)C1 N1(CCC)CC(NC(=O)C(N2CCC(n3cc(Br)cn3)CC2)=O)CC1=O c1(NC(C2CC3(CCCO3)C2)=O)cccc2c1OCC2.CC1(C)CN2CC1C2=O C(=O)(C(C(C)C)n1ccnc1)N(C1CCCN(C2CCCCC2)C1)CC N1(CC)CCCC(C(=O)N(CCCNC(c2csc(C(F)F)n2)=O)CC)C1 C(=O)(CCCC(F)(F)CO)N1CCC(OC)CC1.c12ncc(s1)c(=O)n2C1CC1 c1(OCC)ccc(C(=O)NCC(C)(C)CCNC(=O)C(C)(C)C2CCCO2)cn1 c1(C(=O)NC(C)CCN(C(=O)C(F)=C2CCC2)C)cc(F)c(F)c(F)c1F C(CCC(C)(C)C(=O)NCC(=O)OCC1CC1)NC(C1OCCC(C)C1)=O Cc1nccc(C(N2CCN(C(=O)C(C)NC(N)=O)CC2CCO)=O)c1O CCCCC(C)C(=O)NCc1nocc1C(=O)NC1CC1CN(C)C C1(C(=O)Nc2cc(C(=O)OC)no2)CC2(CCN(Cc3csc(C)n3)CC2)C1 c1(NC(C2CN(Cc3c(Br)ccnc3Br)CCS2)=O)cc(F)ccc1F c1(C(=O)NC(C(C)NC(C2CN(CCCC)C(=O)C2)=O)C)cnc2n1CCOC2 c1(CC)cc(C(N2CCCC(C(N3CCCCC3)=O)C2)=O)cc(N)c1 C1(NC(C(=O)NCCOC)=O)CC2CC(NC(C3(SC)CC3)=O)CC12 C1(CSCC(C(=O)OCCO)OC)CCN(c2ncc(I)cn2)CC1 Cc1cccc([N+](=O)[O-])c1C(=O)NC1CCCN(C(=O)C#CC2CCCCO2)C1 C1(CC)CN(c2ccnc(COC)n2)CCN1C(c1cccnc1Cl)=O CC(C)CC(C)CC(=O)N1CCC(NC(c2cc(O)nc(N(C)C)n2)=O)CC1 C1(NC(C2(CC)COC2)=O)CC12CCN(Cc1c(Cl)cccc1Br)CC2 C(C)(CCCNC(C1(C)CC1C(=O)O)=O)NC(CCNC(=O)OC(C)C)=O C(C(=O)NCC1(c2ccccc2)CCC1)(C1=NOCC1)NC(C(C)NC(C)=O)=O c1(C(=O)NCC2(F)CCC(NC(c3ccc(O)nc3)=O)C2)ccn2ccnc2c1 C1(NC(CCOCCOCC)=O)CCCCC12CCCN(C(=O)CSC)C2 C1(CNC(C2N(C(CNC(=O)OCC=C)=O)CC2)=O)CC1[N+](=O)[O-] c1(C(=O)NCCC2CC(F)CN2)ccc(-n2ccnc2)cc1 CC1CCCC(C2=NOC(C(=O)Nc3cc(Br)ccc3I)C2)C1 C=CC(CC)C(=O)OC(c1cccc(C(C)(C)C)c1)C N1(C(C(C)n2cccn2)=O)CCC(C)(C)C(C(=O)N(C2(CCO)CC2)C)C1 c1(CC)nn(C)c(C(=O)NCCN(C(=O)CCC(C)(F)F)CC(C)O)c1Cl c1(CC(=O)NC(CNC(C(F)OC)=O)C)coc2cc(C(C)(C)C)ccc12 CC1CCCC1(C)NC(c1c(CNC(c2cc(Cl)cn2C)=O)nnn1C)=O N1(C(=O)NCC2(C(=O)OCC)CC2c2cnnn2C)CCC2(CC=CCO2)C1 C1(NC(CC2C(C)CCO2)=O)CCC(C)N(C(c2cc(F)ccc2O)=O)C1 CCCC(CC)CCC(=O)N1CCC=C(CNC(c2coc(SC)c2)=O)C1 n1(C(C)(C)C)ccnc1-c1nccn1NCC(c1ccccc1)CO C1(SC)CCCCC1N=c1[nH]c(N(CCCC(C)C)C)nc2cc[nH]c12 C1(CCC)CN(C(=O)Cn2c(C)ccc2C)CCN1C(c1cc(F)cc(F)c1)=O c1(C(=O)NCCC(C)N(C(CCCn2c(C)ncc2)=O)C)cc(F)c(N)cc1F C1(NC(c2c(CN)cc(N)cc2)=O)CS(=O)(=O)C12CCCC2 c1(C(C)C)ccc(C(=O)NCC2CC(F)CN2C(=O)CCCCC2CC2)nc1 CCC(C)(F)C(=O)NC1CC(=O)N(C2CN(C(=O)Cn3cc(COC)nn3)C2)C1 C1(C(=O)NC(CC=C)CNC(=O)Cc2ccc(C)nc2)Cc2ccc(F)cc2C1 C1(C(=O)NCCCOCCC(=O)N(CC(C)(C)C#N)C)CCCCC(=O)N1 N#CC12CN(C(c3ccc(C4CCCCO4)cc3)=O)CC1CS(=O)(=O)C2 C1(NC(CSCCOC)=O)CN(C(=O)C(COC)OC)CCC12CCC2 N1(C(C2CCN2C(=O)C(c2ccccc2)F)=O)Cc2ccc([N+](=O)[O-])cc2C1 C=CCC(F)(F)C(=O)NC(C)CN(C(=O)C(C)(O)Cc1ccccc1)C N1(C(C(C)C)=O)CCCC1C(N1CC(C)(NC(c2cc(C3CCC3)[nH]n2)=O)C1)=O Cc1cscc1C(=O)NCC1CCN1C(=O)CC1CC=CC1 Cn1cnc2c(N3CC4(CCCN4S(=O)(=O)c4ccsc4)C3)ncnc12 Cc1ccc(CN2CC(C)C2C(=O)Nc2cc(C3CCCCC3)no2)[nH]1 C1(C(N2C(C)C(N(C)C)CC2)=O)N(C(=O)C2=COCCC2)CCCC1(C)C Cc1cc(CC(=O)N(C(C(=O)N(C2CCCC2C)C)C2CC2)C)no1 c1(C(C(N2CCC(NC(C3(OC)CCC3)=O)C2)=O)O)ccccc1Cl c1(C(=O)NC2(C)CCN(C(C34CCCC3CCC4)=O)C2)cc2c(F)cccc2s1 n1(CC)ccc(CC(=O)NC2C(C(=O)NCC(C(C)C)N(C)C)C2(C)C)n1 C1(N(C(c2c(CC)scn2)=O)C)CCC2CN(C(C3CCSC3)=O)CC12 C1(OCCCNC(C2C(c3c(C)nsc3)C2)=O)CCN(C(=O)CC2(C)CC2)CC1 Cc1c(C(=O)N(C)CC2COC(C)(C)O2)sc2[nH]cnc(=S)c12 N1(C(C2CCCN(CC)C2)=O)CCC2(NC(=O)Cc3sc(O)nc3O)CCCC12 C=CCCCCCCCCCNc1ccc(N2CCN(C)CC2)c(Cl)c1 C=CC(CC)C(=O)NCCC1(NC(=O)CC(N2CCCCC2=O)C)CCC1 C1(C2(O)CN(C(=O)CSC3CC3)C2)(CNC(C2CC(=O)N(C3CC3)C2)=O)CC1 C1(C2CCOCC2)(CNC(C2(C)CCC2)=O)CCN(C(=O)CCC2CCCO2)C1 CCCC(CC)C(=O)N(CCC(=O)N(C)CCOCC1CC1)C N1(C(C(CO)NC(N)=O)=O)CCCC(c2ccccc2)(CNC2CC3CCC2C3)C1 C(=O)(C(CC)C(=O)NCC(C)C(=O)NCCc1cocn1)OCC CP(C)(=O)C(O)C(=O)N1CC(CN2CC3CC3C2)C1.n12cc(nn1)C2 C12(CNC(C(C3(O)CCC3)NC(C=C(C)C)=O)=O)CC(C)(CCO1)C2 C1(CC(=O)NCCC2CC(NC(c3c(C)nco3)=O)C2)CN2CCN1CC2 CCC(CC)(CN=C(NC(C)C1CC1)N1CCC(F)(F)C(C)C1)CC c1(C(=O)Nc2nc(-c3cccnn3)n[nH]2)cc(F)cc(I)c1 C1(C(=O)NCC2(NC(COc3ccc(C)cc3C)=O)CC2)CCn2nnnc2C1 C1(NC(c2c(C)nc(-n3ccnc3)s2)=O)CN(C(C2CC2F)=O)CCC1C CC1=CCSC1C(=O)N(CC(O)C(=O)O)C(c1ccccc1)C C1(NC(c2ccnc(Cl)c2F)=O)(CO)CCCN(C(=O)C2=CS(=O)CC2)C1 N1(C(=O)CCSC2CC2)CC2CC1CN2C(C1CCN(S(=O)(=O)C(F)(F)F)C1)=O S(=O)(=O)(c1cccnc1N1CCCC(C)(C)C1)NCC(=O)N(C)C N1(C(CCC2(C)CC2)=O)CCC2(CCCN(C(C3CN(c4nncs4)C3)=O)C2)C1 Cc1ccc(F)cc1CNC(=NCC1C(C)C1(F)F)NC(C)C c1(N2C(CNC(C(CCCOC)C)=O)CC3COCC32)nc2ccc(N)cc2s1 c1(OC(CC)CN(C(C2CCOC2(C)C)C(=O)NCCC#N)C)cccc(Cl)c1 O=C(C#CC1CCC1)NC12CCC1CN(C(=O)C=Cc1ccc(Cl)cc1)C2 CC(CC(=O)NC1CC(=O)N(C)C1=O)C(C)(C)NC(=O)CC(C)(C)C(F)F C1(CN(C(C2C(C)=C2)=O)CC2CC2)CCN(C(=O)CN2CSCCSC2)C12CC2 c1(OC)nccc(C(=O)NC2CN(C(c3ccc(C(F)F)cc3)=O)CC2C)n1 N1(CC(=O)NC(CO)C(=O)NCc2csnn2)CCCCCC1 N1(C(C2(N3CCC(C)CC3)CC2)=O)CC(C(=O)NC2CCCOC2)OC(C)C1 CCCCC(C)CCC(=O)N1CCCC1CNC(=O)Cc1ccc(OC)c(Cl)c1 C=C(C)C1OCCC1C(=O)NCC(C)CN(C)C(c1sccc1C#N)=O Cc1nn(CCC(=O)N(C2(C(C)C)CCC2)CC(C)O)c(=O)o1 C1(C(=O)NC(C2CCCCN2C(c2cc(Cl)ccn2)=O)C)CCCCC1(C)C C1(NC(c2c(C(C)C)n(CCO)nc2)=O)CN(C(c2ccon2)=O)CCC1CO CC1=C(C(=O)N2CC(CC(=O)NCC(C)(C)C)CC2(C)C)CCCO1 C1(NC(C(C)SCCCC)=O)CC2CN(C(=O)Cc3cc(C)ccc3C)CC2C1 N=c1ccc(C(N2CCC(OC3CC3)C2)=O)c(Cl)[nH]1 c1(CC(=O)NC2C(NC(CC=CC)=O)COCC2)cc(C)cc(F)c1 N1(C(CC(CC)CC)=O)CC(C)CN(C(c2coc(Br)n2)=O)C(C)C1 c1(OC)nc(Cl)ccc1C(=O)N(C(C)CCNC(=O)CC(=O)N(C)C)C C(C(C)(C)C#CC(=O)NCCC1CCCCO1)NC(c1c(C)n(C)nc1)=O C1(C(C)C)N(C(c2cscn2)=O)CC12CCN(C(=O)CCC1CCC(C)O1)CC2 c1(C(N(C)CC2(NC(C(C)Oc3ccccc3)=O)CC2)=O)cncc(F)c1Cl c1(OC2CCN(C(CCc3c(C)n(C)nc3)=O)C2)ccc(Cl)cc1F CCCC(C#N)C(=O)NCCCCNC(c1cc(C)ccc1NS(C)(=O)=O)=O C(=O)(CC(C)C(F)(F)F)NC(C(=O)Nc1cccc(OC)c1)CC1CCC1 C1(NC(C(C)(C)n2cncn2)=O)CC2CC1N(C(=O)CCCCCF)C2 C1(N(C)C)CCC(C(=O)NCCn2cc(-c3cc(CO)on3)nn2)CC1 Cc1cc(-c2csc(CNc3ccc(OCCC(C)C)cc3)c2)cc(C)n1 C(CC)(C(=O)N(CCC(C)(C)NC(C1CCC1C(C)(C)C)=O)C)=CC C(CC(CNC(c1cc(CC)no1)=O)NC(=O)COCCOC)OC C1(C(=O)NC2(CCNC(c3cc(CC)no3)=O)CCC2)CNC(=O)CC1C N1(C(C(C)(C)O)=O)CCC(C(=O)NC2CCN3CCC2C3)C(O)C1 C1(C(N2CCC(C(C)NC(c3ccc(C(F)F)o3)=O)C2)=O)CN2CCCC2CO1 O=C1CNC(=O)c2ccc(C(N3CC(NC(=O)CNC(N)=O)C(O)C3)=O)cc2N1 C(=O)(CC1OCc2ncccc21)NCC1CC(C)(C)CN1C(=O)CCCF N1(C(c2cc(C)c(O)nn2)=O)CCC(C)(C)C(C(N2CC3CC2C2CC32)=O)C1 CC(N)(CC(F)(F)F)C(=O)N1CCCC(OC(F)F)CC1 C1(C(=O)NCCC2CCCN(C(C3CC(SC)C3)=O)C2)(CC)CCCCO1 c1(OC)ccc(C)c(-c2cn(C(C)(C)CC(=O)OC3CCOC(C)C3)nn2)c1 C1(NC(c2cnc(C(F)F)nc2)=O)CC2CCC(C1)N2C(=O)CCCF N1(C(CCOCC#C)=O)CC2(CCC(NC(=O)Cc3csc(C)n3)C2)C1 CC(C)CC(C)C(=O)NC1(CC=CC(=O)NC(C)Cc2cn[nH]c2)CCC1 c1(C(=O)NC2CC(NC(c3c(CC)cccc3CC)=O)C2)cc(S(N)(=O)=O)c[nH]1 CC1CN(C(=O)CNC(N)=O)C(C)CN1C(C1CCCCO1)=O N(C(=NCCc1ccc(F)cc1)NCCCS(=O)(=O)N1CCCC1)C1C(C)C1 C(=O)(CC(CN(C)C)CC)N1CC(C#C)(C(=O)NCC(C)CC=C)C1 C1(N=[N+]=[N-])(C(N(CCCNC(=O)CCCn2ccnn2)C)=O)CCOCC1 N1(C(CC2C(=O)NC(=N)S2)=O)CCCC2(NC(=O)Cc3ccc(O)nc3)CC2C1 C(C(CCC)C(=O)NC1CCN(C2CC2)C1=O)NC(c1cc(CCC)[nH]n1)=O c1(C(=O)NCC2CCC(C(N3CCC(CC)C3C)=O)O2)ccc2cc[nH]c2n1 c1(COC)nocc1NC(=O)C(Cc1cc[nH]n1)NC(=O)C(=O)C1CCCC1 c1(C(=O)NC(C2CCOC2)CNC(c2nnc(C)s2)=O)csc2ccccc12 C(c1cn(CC(F)(F)CNC(C2CC(Cl)(Cl)C2)=O)nn1)=CC(C)C N1(C(Cc2cn(C)nc2Cl)=O)CCOC(C)(CNC(c2cn[nH]c2)=O)C1 c1(C(c2n(CCC3(C)CC3)nnn2)N(c2cnccn2)C2CC2)cccc(Br)c1 Cc1cc(Cl)cc(NC(C2CC2C(=O)NC2CCCCC2(F)F)=O)c1Cl CCC(F)(F)CC(=O)NCC1(F)CCC(NC(c2cccc(CF)c2)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CCN(C(C3CCCN3C(=O)C(C)C)=O)C2)C1 C1(NC(c2ccc(C)nn2)=O)CN(C(c2cc(Cl)cn2C)=O)CC2(CCC2)C1 Cc1ncc(C(=O)NCCC2CC(NC(C3(n4cnnn4)CC3)=O)C2)n1C CCC(C)(CCC(C)C)C(=O)N1CCC2(CCCN2C(=O)C=CC(F)(F)F)C1 C1(C(=O)NCC2(CO)CCN(C(C3CC34CC(O)C4)=O)C2)(COC)CCCCO1 C(CCC(O)C(=O)NC(c1cn(C)nn1)C)NC(C=C(C)C)=O C1(NC(c2[nH]cc(OCC)c(=O)c2)=O)CC2CC(C1)N(c1nc(C#N)c(Cl)s1)C2 Cc1c(C(N2CCC(C(C)NC(c3snc(Cl)c3Cl)=O)C2)=O)ccn1C1CC1 c1(C(C(=O)NCC(=C)C)N(C)CCc2ccc(F)cc2)cccc(Cl)c1C c1(C(=O)NCCC2N(C(CN(C)C)=O)CCC2)nc(O)nc(O)c1F c1(C(N2CC(NC(C(C)CCO)=O)CC2(C)C)=O)ccnc2ccc(F)cc12 N1(C(CCCC(=O)OC)=O)C(CNC(=O)C(C)=CC2CC2)CC2COCC12 CCCCC(C)CCC(=O)N1CCC(CC(=O)Nc2cc(OC)ccn2)C1 C1(CNC(c2c[nH]nc2CCN(C)C)=O)C2CN(C(C3C(C(=O)OC)C3)=O)CC12 c1(C(=O)NCCCc2ccc(C)cc2)cc(S(=O)(=O)N(N2CCOCC2)C)c[nH]1 c1(NCCC(=O)NC2(CO)CN(C(C(C=C)O)=O)C2)oc(C)nc1C#N C(CCCCC(=O)NC1C2CCC(C2)C1C(=O)NCc1nnn(C)n1)OC C(=O)(CC(CC)C(F)F)N1CCCC(CCC)(C(=O)NCC(C)(C)C)C1 CCCCCC(O)C(=O)N1CCCC(NC(C2CCC(C3CC3)CC2)=O)C1 c1(OC)cnc(NC(C2(N(C(=O)C(N)=O)C3CC3)COC2)=O)c(F)c1 N1(C(C2C(C(C)C)(CC)C2)=O)C2CCCC1CN(C(C1CC(CCOC)C1)=O)C2 N1(C(C(C2CCC2)OC)=O)CCC(CO)(NC(c2ccncc2N)=O)CC1 N12CC3(CCC(OC3)C1=O)C2.S(=O)(=O)(c1ccccc1)NC1C(OCC)COC1 c1(OC)nc2ccc(C(N3CC(C)CN(C(=O)CSC4CC4)C(C)C3)=O)cc2[nH]1 C(CCN=C(NCc1cnn(CC(F)(F)F)c1)NCC1CCC1)(C(F)(F)F)OC c1(CCC)ccccc1C(=O)NC(C(=O)NC(C)CCN(C)C)C(C)C Cc1cc(C(N2CCN(C(C3CCC(=O)N(C)C3)=O)C(CO)C2)=O)ccc1C#N c1(NC(C2CC(NCc3ccc(Br)cc3Br)C2)=O)cc([N+](=O)[O-])c(Br)cc1F c1(C(N(C(C)CNC(=O)C(C)(C)c2cnco2)C)=O)ccc2nccn2n1 Cc1ccc(-c2[nH]nc(C(=O)NOCC(O)C(F)(F)F)c2C)cc1 C1(CCC)CN(C(=O)CC(C)SC)CC1NC(c1ccc(C)n1C)=O C1(CC(=O)NC(CNC(CS(=O)(=O)NCC)=O)C2CC2)CC2(CCC2)CO1 c1(OC)cc(C(N2CCC3CN(C(=O)CC4(OC)CC4)CC23)=O)sc1S(N)(=O)=O n1(C2CCN(CC(=O)NC3CCC(N)CC3)CC2)cnc2ccccc12 c1(C(C(=O)N(C)C)NC(N)=O)cccc(Cl)c1.c12cn(nn1)CC(=O)NC2(C)C N1(C(c2n(CC)ncc2)=O)CCCOC(CNC(C2(C)CCCCO2)=O)C1 C1(C(N(OC)CC2CCCCC2)=O)CCCN(C(C2C3COCC23)=O)CC1 c1(C(N2CC(NC(c3n(C)ccc3)=O)C3C2C3)=O)cc2c(cn1)OCCC2 Cn1nc(C(=O)OC(C)(C)C)oc1=O.C1(=O)CCO1.C1C(=O)OC(=O)N1 CCC(C(=O)NCC1CCC(F)(CNC(=O)CCn2ccc(C)n2)C1)C(C)C C(=O)(CCCC(=O)NC1CC(C)(NC(=O)CCNC(C2CC2CC)=O)C1)NCC N1(C(C(C)NC(C)=O)=O)CCCCC1CN(C)C(c1cocn1)=O CC1CN(C(=O)CCO)CCN1C(=O)CCSc1ccc(F)cc1 C1(NC(c2ncn(C(C)C)n2)=O)CN(C(=O)CC#N)CC1C C(=O)(C(C)CC(=O)OCC)NC(CC)CNC(c1cc(C(F)(F)F)ns1)=O C1(C(N2CCN(CC#CC)CC2)=O)CCN(C(c2csc(Cl)c2)=O)C(C)C1 N1(C(C(=O)Nc2ccc(OCCC)cc2)=O)CCC12CCS(=O)(=O)C2 C12(CNC(C)=O)CC(C1)C(NC(C1(NC(=O)C3CC3)CC1)=O)CO2 Nc1cc(C(=O)NCC(C)NC(=O)CCC2CCCO2)c2ccccc2c1 Cn1cc([N+](=O)[O-])c(CC(N2CCN(C(C3CCCOC3)=O)C(C3CC3)C2)=O)n1 C1(C(=O)NCC2(COC)CN(C(C3CC(F)(CF)C3)=O)C2)CCNC(=O)C1 C1(NC(C2ON=C(C)C2)=O)CCN(C(=O)CCc2ccc(Br)cc2C)CC1F C1(C(N(CCCC=C)C)=O)CN(C(c2ccccc2)=O)CC1F Cc1cc(-c2ccc(C(=O)NC(c3ccccn3)CO)nn2)cc(C)n1 n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CCC(CN(C)C(C3CC3F)=O)CC2)n1 C1(C)(CNC(c2c(CC)n(CC)nc2)=O)CN(C(C2(C)CSC2)=O)CCO1 C(C)(c1ccco1)=CC(=O)NCCOCC(N1C(C)(CCC)CC1)=O Cc1nc(C=CC(=O)NCCN2CCC(NC(C3CC(Cl)(Cl)C3)=O)CC2)cs1 N1(C(C2(F)C(C)(C)C2)=O)CCC(O)(Cn2cc(-c3ccccc3Cl)nn2)CC1 CCC(C#N)(CC)C(=O)NCC1CN(C(=O)Cc2ccc(Cl)c(Cl)c2)CCCO1 C1(CN(C(C2CC(=C3CCC3)C2)=O)CC)CCCCN1C(c1ccc(C#N)s1)=O N1(CC(=O)OCC)CCCN(Cc2c(C)csc2Cl)CC1 N1(C(C2CCC(C)CC2)=O)CC2CCCC(CNC(c3nn(C)cc3Cl)=O)C2C1 N1(CC)C(=O)CCC1C(=O)NCC1C=CCN1C(=O)C(c1ccc(OC)cc1)=O Cc1ccncc1C1CCN(C(=O)NCc2ccoc2C(F)(F)F)C1 C1(n2cc(CNC(=O)COC(C)C)nn2)CC2CCC1(C(CC)=O)C2 CC(C)C(O)C(C)C(=O)NCC1(C(N2CCCC3(C2)N=N3)=O)CCCC1 C1(NC(CC2OCCN(C(CCc3ccn(C)c3)=O)C2)=O)CCC2(CCC2)CC1 c1(NCCNC(CN(CC)CC)=O)ncnc(OC(C)(C)C)n1 c1(CC(=O)NCC=CCNC(Cn2ncc(C#C)c2)=O)ccc2ccn(C)c2c1 C(=O)(C1=CCC(F)(F)CC1)NC1(C)CC(NC(c2c(C)nc(C)s2)=O)C1 c1(CC)ccc(NC(N(C)Cc2cnc(C(C)O)s2)=O)cc1 Cc1cc(CCC(N2CC3C(C2)C3(F)F)=O)cc(C)n1 c1(C(=O)NC(C)CNC(=O)CP(C)(C)=O)cc2c(o1)CCCC2 CC(C)CCCCC(=O)NC1CN(C2CCC(=O)NC2c2cncn2C)C1 c1(C(=O)NCC(C)C(=O)N(C)Cc2ccon2)cccnc1S N1(C(c2c(O)ncc(SCC)c2)=O)CC(C)CN(C(=O)CCC(=O)NC)C(C)C1 CC1(CC(=O)N(CCCNC(c2ccn(CC(F)(F)F)n2)=O)C2CC2)CCCO1 C#CCC(C(=O)NCC(C1CC1)NC(=O)CC1CCC1)CC(=O)NC1(C)CCC1 Cc1cnc(CC(=O)NC(CNC(=O)Cc2cnc(C)o2)C2CC2)[nH]1 C1(C(N2CC3C(CC)(C3)C2)=O)CCN(C(=O)C2(OC)CCCC2)O1 C1(NC(C2(OCC)CCOC2)=O)CC2CCC(C1)N2C(=O)CC1(O)CCCOC1 C=CC(CC)CC(=O)NC(c1nocc1C(=O)NCC(C)O)C N1(C(C(CC)C)=O)CC2(CNC(C3CSCCS3)=O)CC1CO2 CC1CCOCC1C(=O)NC1CC=CCC1C(=O)NCCC1(C)OCCO1 C1(NC(C=C(C)C)=O)CCN(C(=O)CCC(=O)c2cccc(N)c2)CC1F c1(C(=O)NCC2(F)CC(NC(C3CC4CC4C3)=O)C2)csc2ncnc(O)c12 N1(C(CSCC)=O)CCC(C)N(C(=O)CCc2nnc(S)n2C)CC1 Cc1nc2cc(NC(C3(C)CC34CCN(C(=O)C(O)C(C)C)CC4)=O)ccc2s1 C1(OC)CCN(C(C2(NC(=O)CCCN(C)C)CCC(C)(C)C2)=O)C(C)C1 C=CC(C)(CC)C(=O)N1CCCOC(CCNC(c2c(OC)ccnc2O)=O)C1 c1(C(N(CCCNC(=O)C(C)(C)CF)CC)=O)cc2c(Br)cccc2cn1 N1(C(C(c2ccn(C)n2)C)=O)CC(NC(=O)CN2CCC(O)CC2)C2CCCC12 N1(C(CC2(NC(C(CC)NC(C)=O)=O)CCC2)=O)CCCCC1C1(O)CC1 C1(C(=O)NC(C2CCN(c3ncnc4[nH]ccc34)C2)C)CC(C)(C)CC(C)(C)C1 C1(Nc2cc(C(=O)OC)[nH]n2)CC=CCC1C(=O)OC c1(CNC(C2CC2C(=O)NC(Cc2ccc(F)cc2)CO)=O)c(F)cccc1I N1(C(c2nc(OCC)sn2)=O)CC(CNC(=O)CC23COCC(C2)C3)CC1(C)C c1(CC(N2CCC(O)(CN(C(C(C=C)O)=O)C)CC2)=O)ccc2sccc2c1 c1(C(=O)NCC2(OC)CN(C(=O)CC3CCC(=O)N3)C2)cc2c(O)cccc2[nH]1 C1(NCc2c(C(C)=O)occ2)CCCC(NC(N2C3CCC2CC3)=O)C1.C(C)(C)(C)O c1(OCC)ccc(F)c(C(N2CCN(CC(O)COC)C(C)C2)=O)c1F Cc1ccc(NC(=O)CCC(C)(C)NC(=O)CCC2CCC2)cc1F C(=O)(C(CC(C)C)ONC(C1CC(=O)C1)=O)N(CC=C)C1CC1 Cn1cnc2c(NC3CCCC3C3CC3)[nH]c(=NCC34CCCN3CCC4)nc12 C(=O)(C1c2ccccc2C2CC1C2)NCC(CNC(c1ccc(C)nn1)=O)OC c1(COC)nc(N2CCCCC(NC(C3CC(N(C)C)C3)=O)C2)cc(C)n1 C12(CNC(c3cc(OC)n[nH]3)=O)CCCC1N(C(c1ncc(N)cc1Cl)=O)CC2 N1(C(C(CC)(C)CO)=O)CC2(C=C(C(=O)NCCC(C)F)CO2)C1 c1(C(N2C3(CNC(CCC)=O)CCC3CC2)=O)ccc2[nH]ccc2c1 C(=O)(C(C)(COC)OC)NCC(C1(C)CC1)OC.C1(C)CCC(c2cc[nH]n2)O1 c1(C(N2CCCC(O)(CNC(c3cnon3)=O)C2)=O)ccc(Br)c(F)c1F N(C(=NCCC(C)=O)NC1CCC(C)C1)C1CCN(C(=O)NCC)CC1 C1(C(=O)NC(C=C)C)(CCNC(=O)Cc2nonc2C)CCCC1 C(=O)(C(CC1CCCC1)NC(=O)C(O)CN(C)C)N(CC(C1CC1)OC)C C1(NC(C2CCC(OC(C)C)CC2)=O)CC2CN(C(=O)CC(C)(C)C#N)CC12 C#CC1CN(C(C2CN(C(=O)COCCCF)CC2(C)C)=O)CCO1 N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2(C1)CN(C(C1CC3CCC(C1)O3)=O)C2 C(C1c2ccccc2CCN1C(c1nncn1CC)=O)NC(C(CCC)O)=O c1(C(=O)NC(C)CCCCNC(c2cncnc2)=O)ncc(Cl)cc1Cl C(CN=C(NCC(N1CCC(C)(C)C1)C)N1CCC(n2cc(C)cn2)CC1)OC C1(C(=O)NCCN2CCN(C(Cc3c(C)nn(C)c3)=O)CC2)CCCCC(=O)C1 C(CC(C(=O)NCC1(C)COC(=O)N1)NC(C1CCCSC1)=O)=CC C12CN(CC1C)C(=O)CN2C(CC1CC(C)C1)=O.c1(C(=O)CO)ccc(Br)cc1 C(=O)(C(C)(C)C(F)(F)CC)N1CCC(N(C(c2noc3c2CCCC3)=O)CC)C1 c1(NC=O)ccc(C(=O)NC2CCC(F)(CNC(C3CC4CC4C3)=O)C2)cc1 c1(N2C(C)CC(C(F)(F)F)C2)[nH]c(=NCCC(Cl)=CCl)nc2c1ncn2C c1(C(=O)NC(C)CCNC(=O)CNS(=O)(=O)C2CC2)cc(F)cc(N)c1F N1(C(C23C(CN(C(C4C(C)C5CCC4C5)=O)C2)C3)=O)CC(C)(C)C12CCC2 c1(-n2cc(CC3CCN(C(C(C)O)=O)C3)nn2)ccc(Cl)c(Cl)c1 C12(CC)CN(C(C3CCC=CCC3)=O)C(CNC(C3(OC)CCC3)=O)(C1)C2 c1(CC(N2C(CNc3ccc(SC)cc3)CCC2)=O)cc(F)ccc1F N1(C(CCOCCCOC)=O)CC(O)C(O)C1C(=O)NCC(O)CCSC c1(C(=O)NC(CC)CN(C)C(C2(CO)CCCO2)=O)nnc(S)n1C c1(C(N2CCC(N(C(C3C(C)C3)=O)C)C2)=O)nc2ncc(Br)cc2[nH]1 c1(SC)nc(C(=O)NCCCNC(C23CCCN2CC(O)C3)=O)c2ccccn12 Cc1ccc(F)c(C(=O)NCC(C)(CO)NC(c2ccc(C3CC3)cc2F)=O)c1 c1(-c2scc(NC(C3CCC(O)CC3)=O)n2)c(Cl)cccc1Cl Cc1cc(C(N2CC=C(C(=O)NCCCCCO)C2)=O)nnc1C C1(NC(C2CC(C)OCC2)=O)CC2CC1CN(C(c1ccsc1C(F)(F)F)=O)C2 CCC(O)C(C)C(=O)N(CCNC(=O)C(C)(C)C(C)C)CCOC c1(OC(c2nc(C3CC3)nn2-c2ccccc2C(F)(F)F)CC)ccc(O)cc1 c1(CC(=O)N(C)CC2N(C(C3(C#C)CCC3)=O)CCC2)ccc(Cl)cc1F CCN=c1[nH]cc(C(=O)NCC2CN(C(=O)C(O)P(C)(C)=O)C(C)(C)C2)s1 N#Cc1cc(CC(=O)NCC2(NC(C3C4C5CCC(C5)C34)=O)CC2)ccc1F C(C(CC1CC1)C(=O)N(CCF)CC1CC1)NC(C(N1CCSCC1)C)=O c1(C(=O)OCC)nc(NCCCCC(C)NC(=O)CCCF)c(C)s1 C1(NC(COCCC)=O)CCCC(CNC(=O)CCNC(=O)NC)C1 C=CCCC(C(=O)N1CCC(C(C)OC)CC1)NC(c1cc(C)[nH]n1)=O C1(NC(Cc2cc(C)on2)=O)CCCCC1NC(C1CCCCS1)=O N1(C(=O)Nc2nnc(-c3ccc(F)cc3)s2)CC2CC(C1)C2(F)F C=CC(CCC)CC(=O)N1CCC(CN(C)C(c2cc(C3CC3)ncn2)=O)C1 Cn1nc(Br)nc1C(c1nnnn1C(C)(C)C)NCC1(c2cccs2)CC1 c1(C(N2CCC(OCC(F)F)CC2)C(=O)NC(CC)C)c(C)nn(C)c1Cl c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CCC2)cccc2c1OCCCO2 c1(C(N2C(CNC(C(C)OCC=C)=O)CC2)=O)coc(C(C)OC)n1 Cn1nc(C(N2CC3CN(C(=O)Cc4ccsc4)CCC23)=O)c2c1CCSC2 Cc1cccc(C(NOC)=O)c1O.N12CCC(C13CC3)C2=O.N1(C=O)CCOC1 N1(C(C(CCCC)O)=O)CCC2(CC1)CC2NC(C1CCC(=O)N(CC)C1)=O C1(C)(C(=O)NCCC(C)NC(C2CCC(C)O2)=O)CCS(=O)(=O)CC1 Cc1cc(C(N2CCN(c3ccnc(C4CC4)n3)C(C)C2)=O)nc(C)c1 CC1CC(C)(C(N2CCCC2CNC(c2cnc(Cl)c(C3CC3)c2)=O)=O)CCO1 Cc1cc(C)c(C(=O)NCC(C)(C(C)C)NC(c2cc(C#N)c(C)s2)=O)c(O)n1 Cc1cccc(C(=O)NC(C)C(=O)NC23CC(C2)N(C(=O)CC2(O)CCC2)C3)c1 N1(C(c2c(CC)nns2)=O)CCC2(CC1)CC2NC(=O)C(CC)SC CCC(C)CCC(=O)NCC1CC(C(=O)N(C2CCOC2)CC)=NO1 N1(C(Cn2cnc(C)c2C)=O)CC(C)(C)C(O)C1(C)C C1(NC(C2CCN(Cc3ccccc3)C2)(C)C)CCOCC1(C)C c1(CN2CC(C(=O)Nc3cn(CC)nc3C)C2)c(Br)cc(F)cc1Br c1(CCNC(CNC(C)(C)C)=O)nncn1COc1ccccc1.C1CC(=O)O1.O.C.O C(=O)(C(C(C)C)NC(c1ccccc1F)=O)N1CC(C)(OC)C1 c1(OC)ccc(Cl)cc1-n1nc(CC(C)C)nc1C1COC(=O)C1 C(CC)(C(=O)NC1(C(=O)NC(C)(C)CCN(C)C)CC1(C)C)OCC C1(C)(C(N2CCC(C(C)NC(=O)C(C)n3cccc3)C2)=O)CCS(=O)(=O)CC1 C1(CC(=O)NCC2C(CNC(c3c(Cl)cn(C)n3)=O)CCC2)CCC(=O)NC1=O C(=O)(C1CCSc2ccccc21)NCC1(F)CCC(NC(=O)Cc2ccno2)C1 N1(CC)CCN(CCC(=O)NCC(O)CN(C)C(C2CCCS2)=O)CC1 O=C1OC2CON(C(=O)c3cc(-n4cccn4)ccn3)CC2O1 c1(NC(=O)NC2CC(c3cn(C4C5CC6C(C5)C46)nn3)C2)cc(F)cc(F)c1 CC(C)CC(C(=O)N1CCN(C)C(CNC(=O)CC2CC(=O)NC2=O)C1)C(C)C S(=O)(=O)(c1cnc(C)c(C#N)c1)NC(c1cccc(Cl)c1)CC c1(C(C(=O)N(C2CCC(O)C2)C)(C)C)ccc(Cl)cc1 C1(CN(C)C(C2CC23CC3)=O)CCN(C(c2csc(Br)c2)=O)C1 C1(C(=O)NC2CCCC(C(=O)NC3CCOC34CCC4)C2)CC2CCC1CC2 CC(CC(=O)N(CCCN(C(=O)C=C1CCSCC1)C)C)C1CCCO1 c1(NC(C)=O)cccc(-c2nc(CC3CCS(=O)(=O)C3)n(C(C)C(F)(F)F)n2)c1 C1(NC(=O)COCc2ccccn2)CC2(NC(=O)Cn3cnnn3)COC1C2 C(C)(CO)(C(=O)NCCC(C)(C)CNC(=O)Cc1csc(C(C)(C)C)n1)OC c1(CCCC)ocnc1C(N1CC(CO)(NC(c2csc(=N)[nH]2)=O)C1)=O C1(C(=O)OCC)CC(F)(CF)C1.c1(C2C(=O)N2)ccccc1 C1(C(=O)NCCNC(C2(OC3CCCC3)CCOCC2)=O)(OC)CCCCCC1 c1(CC)ccc(C(=O)NCC2CN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)c(O)c1 N#Cc1ccc(=NCC(=O)N2CC3(CCN(C(C4(CF)CCC4)=O)C3)C2)[nH]c1 CCCC(O)CC(=O)N1CC2CC(CNC(=O)CCn3nc(C)cc3C)C2C1 n1(CC)nc(C)c(C(=O)NCC2CC(NC(C3NC(=O)CC3C)=O)C2)c1C C(=O)(C1=CC2CCCC12)NCCN(C(=O)C(C)NC(=O)NC1CCCC1)CC c1(C(N(CCNC(CCC=C=C)=O)CCOC)=O)ccc(CC)c(N)c1 C1(CC)CN(C(c2ccccc2Cl)=O)CCC1NC(=O)CSc1cccc(C)c1 n1(CC)nnc(C)c1C(=O)NCC(C)NC(c1cnoc1-c1ccccc1)=O C1(CCC)CN(C(=O)C(C)CC(N)=O)CCN1C(=O)CCc1ccc[nH]1 C(=O)(C(F)(F)C(F)F)NC(CCN(C(C(C)(C)NC(=O)NCC)=O)C)C1CC1 c1(C(=O)NCCC2(NC(C3C(C)CN(C)C3)=O)CC2)csc2cc(Cl)cnc12 C(=O)(CC(C(C)C)c1ccc(F)c(C)c1)N1CC(N(C(CC2(OC)CC2)=O)C)C1 C1(COC)CN(C(=O)COCCF)CCN1C(c1cnnc(O)c1)=O CCC(CCC(=O)NC(C)(CNC(c1cc(C)cc(C)n1)=O)C1CCC1)OC C(C(CC(C)C)OC)NC(C(CC)NC(c1ccc(CO)cn1)=O)=O C12(c3sc(C(=O)OC)c(C)n3)CCN(CC1)C(=O)N2CC.S(=O)(=O)(C(C)C)NC S(=O)(=O)(c1ccc(C#N)c(NCc2cnc(C)s2)c1)N1CCC(CC)C(C)C1 CCC(C)(C)C(c1nnnn1Cc1cccs1)NCc1cc(N(C)C)no1 C1(C(CNC(=O)CCCc2nccs2)F)CCN(C(=O)CCOC2COC2)CC1 C=CCC(C(=O)NCC=CCNC(c1occc(=O)c1OC)=O)C(C)C Cc1ccc2c(=NCC3(NS(C)(=O)=O)CCCC3)[nH]c(=NC3CCCC3C)[nH]c2c1 C1(C(N(CCNC(CC=CC)=O)CCSC)=O)CCCCN1CCC C(=O)(CCS(=O)(=O)N1CCOCC1)NC(C)CN(C)C(C1(C2CCC2)CC1)=O c1(C(C(=O)NCCOCC2CC2)N(C)CC)ccc2ccc(Cl)cc2n1.C(C)(C)(C)O N1(C(CC=CCC)=O)CCC2CCCC12C(N1CCC(CN(C)C)C1)=O CC(C)CC(=O)NC(C(=O)NCC1C2COCC12)C1CCC1 C1(NC(CSCCC(C)C)=O)CC(O)CN(C(c2ccnc(N(C)C)c2)=O)C1 S(=O)(=O)(c1ccc(NCc2cn(CC3CSC3)nn2)c(Cl)c1)NC(C)C Cc1cc(C(=O)NC(C2CCCN(C(=O)C=CCO)C2)C)cc(O)c1 c1(C(N2CC(N(C)C(c3ncn(C)n3)=O)C(F)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 C1(CNC(C2(C(N)=O)CC2)=O)CCN(C(c2nn[nH]c2Cl)=O)C12CC2 c1(OCCSNC(c2nc(=O)o[nH]2)C)cccc2c1OC(C)(C)C2.O N1(C(CCc2n(C)cnc2)=O)CCC(NC(=O)C(F)=C2CCC2)C(O)C1 Cc1cc(C)c(-c2nc(C3CC3)nn2C2CCOC(C)C2)[nH]1 Cc1c[nH]c(CC(N)=O)c1C(=O)NC1CCC1NC(c1n[nH]cc1Cl)=O O=C(C(O)CC1CCCC1)NCC1(NC(C2(C(N)=O)CC2)=O)CC1 n1(CC)c(N2CCC(F)(NC(=O)OC(C)(C)C)C2)nnc1-c1sccc1O c1(C(=O)NC(CC=C)CO)nc(CNC(=O)C(CSC)OC)oc1C Cc1noc2cc(C(N3CC(NC(=O)C4CC4)C(C)C3)=O)ccc12 C1(NC(C2C(C)C2)=O)CN(Cc2cn(-c3ccc(F)cc3)nn2)CCC1C C1(CNC(C(C)NC(=O)NC)=O)CCN(C(c2cnn(CCO)c2)=O)C(C)C1 C(=O)(C(O)C(C)(C)C)N(CCNC(C1(C(=O)OCC)CC1)=O)C CCCC(CC(=O)NCc1ncccc1O)NC(=O)C(O)CC N1(C(c2ccc(C(=O)OC)nc2)=O)CCN(C(c2cc(C)co2)=O)CC(O)C1 c1(C(=O)NCCCN(C(c2c(C)cc[nH]c2=N)=O)C)ccc2nc(O)n(C)c2c1 C(=O)(C1CCOc2ccccc21)NCC1(F)CC(NC(C2N(CC)CC2)=O)C1 c1(C(=O)NCC2(O)CCN(C(c3c(CCC)onc3C)=O)C2)coc2c1COC2 N1(C(c2ncc(CC)nc2)=O)Cc2nccn2CC(NC(=O)CC2C=CCC2)C1 N1(c2ccc(C(N(CC(N)=O)C)=O)cn2)CC(=O)C2(CCCCC2)C1 N1(C(C(CC)N(C)C)=O)CCC(CNC(c2ccc(-c3ccco3)[nH]2)=O)C12CC2 c1(OC)ccc(F)cc1C(=O)NC1CN(C(C2CN3CCN2CC3)=O)C1 c1(C(=O)NC(CNC(C2OCC(C)C2)=O)C)cc2n(n1)CCCC2O N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C(c2nc(C)ccc2F)=O)CC1CCO N1(C(C(CC)=CC)=O)CCC2(CC1)CC(NC(=O)Cc1cncn1C)CO2 N1(C(C(Cc2ccccc2)C(=O)Nc2ccccc2)=O)CC2(NC(=O)CO)CC1C2 c1(C(N2CC(OCCNC(=O)C=Cc3nccs3)C2)=O)ncc2ccccn12 C=CC(CC)CC(=O)C(N1CC(C(=O)ON2CCCCC2)C(C)(C)C1)=O N1(CC(N2C(C)CCCC2)=O)CCC2(CC1)CN(C(C1CCCN1C)=O)C2 n1(C(C)(C)C)ncc2c(N3CCCC(NC(=O)C(O)c4ccsc4)C3)ncnc12 C(=O)(C(C)S(N)(=O)=O)N(C)CC1CCN(C(C=C(CC)CC)=O)C1 CC(C)CC(C(=O)N1CC2CCOC2(CNC(=O)C#CC2CC2)C1)C(C)C C1(C)(NC(C2N(C(C)C)C(=O)CC2)=O)CCCN(C(C23CCCC2C3(F)F)C)C1 c1(NC(c2nccn2-c2ccccc2)C)nccc(=NC2CCCC2F)[nH]1 N1(C(=O)CC2C=CCC2)CC(C2CCN(C(c3cnc4sccc4c3)=O)CC2)C1 C(=O)(C1Cc2c(Cl)cccc21)NC(CNC(c1ccc(OC)cc1)=O)(C)CO c1(NC(C)(C)C)cccn(C)c1=O.c12ccc(cc1)OC(=O)N(C)C2 N1(C(C2(C)CCCN(C(=O)NC(C(=O)OC)C)C2)=O)CC(C)OCC(C)(C)C1 N1(C(c2ccc(CNC(Cc3ccc(C)nc3)=O)cn2)=O)CC(C)CC(O)C1 CCCCC(F)C(=O)NCc1cc(C(=O)NCC2CCCC2O)n(C)n1 CC(C(=O)NC(CNC(=O)CC1CC2(CCO1)CC2)C1CCC1)C(C)(C)C c1(OC)cccc(SCC(N2CC(N(C(=O)CSC(F)F)C)C(O)C2)=O)c1 N1(C(C)=O)CCC2C1CCN2C(=O)CCNC(C1CCC1)=O C1(CNC(C2CC2(F)F)=O)(NC(C2(CO)CC2)=O)CCOC1 c1(OC)ccc(F)c(C(N2CC(CNC(C3C(C)C3C)=O)CC2(C)C)=O)c1 CCC1=NOC(CC(N2CC(CC(F)C(=O)NC(C)(CC)CC)C2)=O)C1 C(=O)(C1=C(C)C(C)(C)OC1=O)N1CCCC(CCNC(C2(C)ON=C(C)C2)=O)C1 C1(CNC(CCN(CC)CC)=O)C(C)CCCN1C(c1nnc(O)cc1O)=O c1(C(=O)NCC(C=C)O)occc1CNC(c1ccnnc1)=O N1(C(=O)OC(C)(C)C)CCn2c(cnc2C(=O)Nc2cc(C(N)=O)ccc2Cl)C1 C1(C(=O)OCCCCCCCC)CN(C(=O)CC)c2ccc(F)cc2O1 c1(CC)cnccc1CNC(=O)NOCCF CCCCCC(O)C(=O)N1CC2(C(N3CCC(CCO)C3)=O)CCC1CC2 C#CC1CN(C(=O)C(CC=CC)NC(=O)CCC2CCOC2)CCN1C C1(CCC(=O)NC(CC(=O)OCC)C)CCCCN(C(C2CC(=O)N(OC)C2)=O)C1 N1(C(CC2CC(=C)C2)=O)CCC2(CC1)CN(C(c1ncncc1Cl)=O)CC(C)O2 C1(C)(CNC(C(C)Cc2cnn(C)c2)=O)CCCN(C(=O)C2=CCSC2)C1 C1(NC(C(C)OCC)=O)CC(F)CN(C(c2cc(Cl)n(C)n2)=O)C1 C=C1CCN(C(=O)CCN(C)CCN(C(=O)C(CC)n2cncn2)C)C1 c1(-c2cccc(SC)c2)cnc2c(C(=O)NCC3CCCOC3)c[nH]c2c1 c1(C(=O)NCCC2CN(C(C3CN(C)C3)=O)CC(C)O2)cccc2nccnc12 c1(C(N2C3CC(CC(NC(C(C)S(N)(=O)=O)=O)C3)C2)=O)cn2cc(F)ccc2n1 CCCC(C(=O)N1CCC(CF)(NC(C2CCC3(CC2)N=N3)=O)C1)S(N)(=O)=O N1(C(c2nc(C(C)=O)sc2)=O)CC(NC(=O)C(F)(F)c2ccnn2C)CC1C Cc1[nH]c2ncccc2c1C(=O)N(CCNC(=O)Cc1cc(CO)on1)C(C)C C1(CNC(c2ccc(F)cn2)=O)CC12CCN(C(=O)C(O)Cn1cncn1)CC2 c1(C(N(C)CCNC(c2cc(F)c(Br)cc2F)=O)=O)cc2c(=O)[nH]ccn2c1 Cc1nc(C(=O)NCC2(O)CN(C(C3CC4OC3C3CC43)=O)C2)c2ccnc-2[nH]1 C1(NC(c2nc(C)oc2)=O)CC2CCC(C1)N2Cc1nnc(C(C)(C)C)o1 N(C(=NCCN1CCCC1)NCC)C(C)Cc1ccccc1.c1(N)cccc[n+]1[O-] CC1C(C(=O)NC(C)(C)CCn2ccnc2)CCN1C(C1CCC(C)(C)C1)=O C(=O)(CC(C)(C)CNC(c1ccn(C)n1)=O)NC(COC)CCO CC(C)(C#CC(=O)N1CC(OCC(F)F)C1)COC(=O)C=CC(F)F Cc1cc(NC(=O)CC2COCCN2C(=O)C(O)C(C)C)cnc1Cl C=CC(C)(CCOC)C(=O)NCC1(C)CC(NC(=O)COc2cc(C)on2)C1 N1(c2cc(CC)ncn2)CCOCC(NC(c2c(C(F)(F)F)coc2C)=O)C1 c1(CC)ccc(C(N2CCCC2CCC(=O)NCCn2cc(C#N)cn2)=O)cc1 c1(C(=O)NCC2=CCN(C(CN3CC(C)(C)C3)=O)CC2)ccc2c(c1)C(=O)NC2 C1(O)(C(=O)NCCCc2onc(C)n2)CCN(C(=O)OC(C)(C)C)C1 c1(CC)nncn1NC(=O)C1C(NC(=O)COCc2cccnc2)C1C C1(NC(C(C(=C)Cl)(C)C)=O)CC1C1CCN(C(c2cc(C3(C)CC3)on2)=O)CC1 c1(C(N2CC(NC(c3n(C(C)C)ncn3)=O)C(O)C2)=O)c(O)cccc1Cl C=C(C)CC(C(=O)NC1CC(CCNC(=O)CC2CCCC2O)C1)OC N1(C(Cc2scc(C)c2)=O)CC(F)CC1CC(=O)NCC(N1CCOCC1)C c1(CC)oc(C)cc1C(=O)N(CCCCCCNC(C1CCC1C(=O)OC)=O)C C(C(CC(=O)NC1CCOCC1C)C1CCC1)NC(C(C)C#N)=O N1(C(C2C(CC)C2)=O)CCC2(C(=O)NC3CC3CC)CCCC12 C1(CC(=O)N(CCCO)CCC)CCCN(C(c2nnc(S)n2C)=O)C1 C1(N(C(c2[nH]cc(C)c2)=O)C)CN(C(=O)C(C)OCC2CC2)CCC1C Cc1noc(C)c1C(C)C(N1CC=CC1CNC(C1CCOC1(C)C)=O)=O N1(C(C(C)(C)C2CCC2)=O)CC2(C1)SCCC2NC(=O)COCc1cccnc1 CCC(CCOC)C(=O)NCC1CN(C(c2ccnn2COC)=O)CCN1C N1(C(CSS(C)(=O)=O)=O)CC(CNC(c2cnc(-c3ccco3)s2)=O)C2CC12 c1(OCC(N2CCN(C(c3cnc(C)o3)=O)C(CF)C2)=O)c(C)cc(Cl)cc1C C(=O)(C(O)(C(F)(F)F)C(F)(F)F)N(C(c1c(C)cc(NCC2CC2CF)s1)=O)CC N1(C(c2c(C)cc(F)c(N)c2)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C2CCCC12 C1(=CC(=O)NCCN(CC(C)O)C(=O)COC2(C)CCC2)CN2CCC1CC2 N1(C(C(C(=C)Cl)(C)C)=O)CC2CCCC2(NC(=O)CCC)C1 Cc1cc(C(=O)NCCC2CN(C(C3CCC3(C)C)=O)CCO2)n2ncnc2n1 CCCC(C#N)C(=O)N1CCN(C(=O)CN(C)S(N)(=O)=O)C(C(C)C)C1 c1(C(N2C(CC)CN(C(=O)CC3CC(F)C3)CC2)=O)cc2c(s1)CCCNC2=O N1(C(CCOC)=O)CCN(C(=O)C(CN(C)C)N(C)C)CC1CC1CC1 Fc1cccc2c1OCC2N=c1nc2scnc2c(NCCC=CBr)[nH]1 C(=O)(C(C)(CO)CO)N1C(C(=O)Nc2ncn(C)n2)CC1 C1(C(N2CC(C(N)=O)(OC)C2)=O)C2CC3C(C2NC(C2(C)CCCCC2C)=O)C13 c1(C(N2C3CN(C(=O)Cc4ccsc4Br)C(C3)C2)=O)n[nH]c2c1CCCC2 C(Cc1ccsc1)(CC(=O)O)NC(c1n(C)cnc1)c1nnnn1C C1(C(=O)NC2(CCNC(C(C)(C)F)=O)CCC2)CC(=O)CC(=O)C1 c1(N2CCC(NC(c3cc(C)no3)=O)C2)cc(CC(C)C)ncn1 C1(C(=O)NCC(C(C)C)NC(c2csc(-c3ccsc3)n2)=O)CC(C)(C)CN1C C(=O)(CCCCC(C)C)NCC1(CCNC(c2ncc(OCC)nc2)=O)CC1 Cc1cccc(Br)c1OCC(N1CC(n2cc(C3CCCOC3)nn2)C(C)C1)=O c1(C(=O)NCC2CN(C(COCC)=O)CC2C)ccc(C#N)cc1 c1(C(=O)NCCCC(C)NC(C(CC(=O)OC)(C)C)=O)ccc2c(c1)SCCN2 c1(C(=O)NCC(C)(CO)NC(C(C)OCCOC)=O)ccc(-n2ccnc2)cn1 N1(C(CCn2ccc(C)n2)=O)C2CCCC1CN(C(C1CCCNS1(=O)=O)=O)C2 c1(OC)cn(CC(=O)NC2CCCCCCN(C(=O)CCOC)C2)c(C)cc1=O C1(CN(C2CCN(S(C)(=O)=O)C2)C)CN(C(=O)Cc2ccc(Cl)cn2)CCO1 C1(CC=C)CCN(C(C2CCCN2C(C2COCCO2)=O)=O)C1 c1(C(=O)NCC(C)NC(C(CCCCCC)C)=O)nc2ccc(CO)cn2c1N C1(C=C)(C(=O)NC(C(=O)NC(CC#C)C(=O)OCC)CCF)CCOCC1 N1(C(C(CC)C)=O)CC2CCCN(C(=O)CCc3ccsc3Cl)C2C1 C(C)(CCCCNC(C1(CN(C)C)CC1)=O)NC(COCC(C)C)=O c1(C(=O)NC(C(=O)NC(CCCCC)C)C(C)(C)C)c[nH]c2ccccc12 N1(CCC(=O)N(C(C)CNC(C2CC2CC(C)(C)C)=O)C)CCCCC1.C1CS1 N1(C(Cc2nc(CC)sc2)=O)CC(NC(c2ccc(Cl)cn2)=O)C(C)(C)C1 c1(C(N2CCC(NC(CN(CC)CC)=O)(CF)C2)=O)c2c(nn1C)CCCC2 N1(C(CCc2c(C)nccc2)=O)CCN(C(=O)C(C2CCOCC2)C)CC1CO c1(C(N2CCCN(C(CC(CC(C)C)C)=O)C(C)C2)=O)cccc2oc(O)nc12 CCC(O)CC(=O)N1CCC(O)(C(C)NC(C2CC2F)=O)C1 CC(C)(CCCNC(=O)Cn1cc(CO)nn1)C(=O)NCC1CNC(=O)CO1 N1(C(CCOCCC)=O)CCC(C2CC2)C1C(=O)NC1CC(C)(N(C)C)C1 N1(C(c2nc(C)oc2)=O)CCC(NC(=O)CC2CC2C(F)(F)F)C(C)C1 C(C(Cl)C(C)(F)F)N(C(=O)CCCn1cc(C2CC3CC3C2)nn1)CC=C c1(C(N(C2CCN(C(C(C(CC)O)C)=O)C2)C)=O)ccc2nc(C)nc(O)c2c1 c1(C(=O)NCC(CCNC(C2(CC=C)CC2)=O)O)cnc(C(C)(C)C)nc1C C(=O)(C1=NOC2(CCC2)C1)N1CCCN(C(CC(CCSC)O)=O)CC1 C(=O)(C(C(C)C)c1cccnc1)NCC(C1CC1)NC(c1n(CC)ccc1)=O c1(C(N2CCN(C(c3c(C)cns3)=O)CC2CCO)=O)cnc2[nH]nc(O)c2c1 c1(C(=O)OC)cc(OC)c(S(=O)(=O)N2CCCC(C3CCCC3)C2)c2ccccc12 c1(SCC(=O)NC2CCN(C(c3cc(C(N)=O)no3)=O)C2)ccccc1Cl C1(C)(CNC(CCn2ncc(C)c2)=O)CN(C(C2(O)CC2(C)C)=O)CCO1 c1(C(C)C)ccc(O)c(C(N2CCC(NC(=O)Cn3cnnc3O)C(C)C2)=O)c1 N1(C(C2CN(C)C2)=O)CC2(CC(C(=O)NCC(O)C(F)F)CO2)C1 c1(OC)ccc(C(N2CC3CC(C2)N3C(=O)CC2CCN(C)CC2)=O)c(Br)c1 C(C(C)(C)CC(=O)OCc1ccc(C(C)(C)C(F)(F)F)cc1)OC N1(C(C(CC2CCC2)OC)=O)CCC(F)(C(N2CCCCC2C2CCC2)=O)CC1 C1(O)(CNC(CCN(C(C)=O)C)=O)CCCN(C(c2ccccc2CC#N)=O)C1 N1(C(c2cccc(C#C)c2)=O)CCC2CN(C(=O)C=Cc3cn(C)cn3)CC2C1 N12CCC3(COC(C3)NC1=O)C2.c1(C(=O)NC(C2CCCC2CO)C)cccn1C N1(C(C(COC)N(C)C)=O)CC2(C1)CN(C(c1ccnc(C3CCC3)c1)=O)C2 c1(C(N(C)CC2(O)CCN(C(C3CC3F)=O)CC2)=O)cncc2cc(Cl)ccc12 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(F)Cc2ccccc2)C1(C)C c1(C(=O)Nc2cc(F)cc(OC)c2Br)ccc(B(O)O)c(Br)c1 N1(C(c2cc(CC)no2)C(=O)NC(C)C)CCCC(c2noc(C(C)C)n2)C1 C1(CC(=O)NC2(CNC(c3scc(COC)c3)=O)CC2)CCc2sccc2C1=O C1(C(=O)O)(NC(C2(NC(=O)OC(C)(C)C)CCSC2)=O)CCCSC1 C1(OC)(CNC(=O)C(C)Sc2ccccn2)CN(C(=O)C(c2ccn(C)n2)C)C1 Cc1n[nH]c(C)c1C(N(C(C1N(c2ncccn2)C(C)CC1)=O)C1CC1)C1CC1 CCCC(CC(=O)N1CCCC(C2OCCO2)CC1)C1CCC1.C1CO1 c1(C(N2C3C(NC(=O)C=Cc4cccc(Cl)c4)C(C3)C2)=O)cc2cccnc2o1 c1(C(N2CC(C(=O)NC(c3c(OC)cccc3)C)C2)=O)ccc(C)nc1C C1(C(=O)NCC2CCCS2)CCC2(CC2)N1C(C1(Cl)CC1(F)F)=O C1(F)(CNC(C=CC(=O)N(C)C)=O)COCCN(C(C2C3(CC3)C23CC3)=O)C1 N(S(=O)(=O)N(C)Cc1csc(C(C)Oc2ccccc2)n1)CC(=O)OC c1(CC(N2CC(NC(C(c3ccccn3)C)=O)C2)=O)ccc(Cl)nc1 c1(OC)cc(C(N2CC(NC(=O)C(C)(F)F)CC2C)=O)c(N)cc1F CC1COCC(C(N2CCOCC2CNC(c2ccnc(C(N)=O)c2)=O)=O)O1 c1(C(C(N2CC(COC)(CNC(=O)CCSC)C2)=O)N(C)C)ccccc1Cl Cc1cc(Cl)ccc1NC(=O)CC1CCCCC1NC(=O)CCN1CCCCC1 c1(C(N(C2C3CN(C(C(CSC)(C)C)=O)CC32)C)=O)coc(=O)c2ccccc12 c1(C(N2CC(CNC(CCNC(=O)NC)=O)C2)=O)cnc(O)n1CC N1(CC)CC(C(=O)OC(C)(C)C)CC(CC)C1.C1C(C)(O)CNC(=O)N1 c1(C(N2CC(NC(CCC(C)OC)=O)C(n3ccnn3)C2)=O)cnn2ccsc12 N1(C(C2(C(=O)OCC)CC2)=O)CC(NC(C2CCCC(OC)C2)=O)CC(O)C1 C1(CC=C)(C(=O)NC(CC(=O)NC(C)(C)C)C2CC2)CN(C(c2nc[nH]n2)=O)C1 C=CCC(C)(C)CC(=O)NC1CC2CC(C1)N(C(c1cn3ncccc3n1)=O)C2 N1(C(CC)=O)CCC(C2CCN(C(c3cnn(CC(F)(F)F)c3)=O)C2)C1 C1(C(=O)NC2(CCNC(C(C(C)C)C3CCC3)=O)CCC2)COCC(C)(C)O1 CCC(CC(=O)N1CCCCC1C1(NC(c2onc(Br)c2C)=O)CC1)C1CC1 C1(C(N(CCCOCCN)C)=O)CCCCNC1=O.C(C(C)(O)C=O)OC N1(C(C2C(CCOC)C2)=O)CCC(C)(CNC(=O)CC2CCCS2(=O)=O)CC1 C(CC(C)(C)NC(=O)OC(C)(C)C)NC(N(c1ccncc1)C(CC)(C)C)=O C1(CC(=O)NC(C(C)NC(CCCOC(C)C)=O)CO)C=NN(C)C1=O CN1CCC(F)(CNC(=O)C(CCC2CC2)NC(c2cc(CO)n(C)n2)=O)C1 C1(NC(=O)CCc2ccoc2)CCC12CCCN(C(=O)CC(F)(F)C(F)(F)F)C2 Cc1coc(C(N2CCC(C3CCCN3C(c3ncc[nH]3)=O)C2)=O)c1 N1(C(C(CC)(F)F)=O)CC(C2CCN(C(C3(CO)CCCCO3)=O)CC2)C1 c1(C(N(C2CC(NC(c3ccc(F)o3)=O)C2)C)=O)ccn(CC(F)F)c(=O)c1 c1(CC(=O)NC(C)CNC(=O)C=CCO)csc(-c2ccccc2)n1 C(=O)(CCCCN1CCCCC1)NC1C(CNC(Cc2n(C)ccn2)=O)CCC1 N(C(=NCCSC)N1CCCC(C(=O)NCC2CC2)C1)c1ccc(CCC)o1 CC1CCCCC1CNc1cc(-n2cccc2)ccn1 CC1CN(C(c2nncs2)=O)CC(C)CN1C(c1cc2ncccc2[nH]1)=O N1(C(c2cc(-c3ccc(C)s3)on2)=O)CCc2nc(=N)[nH]cc2C1 C1(OC)CC(C(=O)NC(C)(CNC(=O)CCc2cnc(C)s2)C2CC2)CC1OC C1(C(F)(F)F)(C(N2CC(CCCCNC(COCC#C)=O)C2)=O)CCCCC1 CC1(C)CC(C(=O)NCCNC(c2c[nH]cc2Br)=O)CC1(C)C c1(CN(CCCCCC)C(=O)Cc2nnnn2C2CCOCC2)cc(F)ccc1F c1(C(=O)NC2(CNC(C(CC)C#N)=O)CCOC2)cccc2c1CCCC2 c1(OC)cccc(C)c1.C1(C(=O)OC)(C(C)C)CCCN1C(=O)Cn1c(C)ccc1C C(=O)(CS(=O)(=O)CC(=O)OC)N1C2CCC(NC(C(C=C=C)C)=O)(CC2)C1 O=C(C#CC1CCOC1)NC1CC2CC1N(C(=O)C1=CCCC1)C2 C1(F)(CNC(C(C)(F)F)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1 c1ccc(S(=O)(=O)CCn2c(-c3cccc(C)c3C#N)ncc2)cc1.N(C)C C1(CNC(c2cc(CNC(N)=O)c[nH]2)=O)C=CCN1C(c1ccon1)=O.N Cc1ccc(S(=O)(=O)N(CC(=O)NC23CCC(C2)C3)C)cc1.C12CCN(C1)C2=O c1(OCCOC)ncc(CNC(c2cc(F)ccc2F)CF)cc1Cl CCC(CO)N(C(=O)C=C(C)CN(C(=O)CC1CC(N(C)C)C1)CC)C C1(Cn2cc(C(C)NC)nn2)CCN(C(c2nc[nH]c2C(F)(F)F)=O)CC1 N#Cc1ccccc1C(=O)NC1CCC1NC(c1ccc(Br)c(Cl)c1)=O N1(C(CNC(=O)NC)=O)CCCC(O)(CNC(C2(CF)COC2)=O)C1 N1(C(C2CCC(C)O2)=O)CC2(NC(=O)CCC(C)(C)F)CCC1CC2 C1(NC(c2c(C(=O)OC)[nH]cc2)=O)CCCC(NC(C2CCCS2)=O)C1 c1(C(=O)NC(C)(CNC(C2CC=CCO2)=O)CO)cccc2ccoc12 C1(CC(=O)NC2(c3ccn(C)n3)CC2)CCCN(C(C2(C(F)F)CCC2)=O)C1 Cc1csc2ncnc(N3CC4(CC4)CC3C(=O)Nc3ccc(Br)nc3)c12 CC1(C)CCCN(C(c2cc(C3CCC3)on2)=O)C1CNC(C1CCCC1O)=O CC(C)C(CC(=O)NC1CCSCC1)NC(c1cc(C#N)cn1C)=O C1(CC=C)(NC(=O)CCC#CC)CCN(C(=O)CSC2CCOC2=O)C1 C1(NC(C(CC2CC2)OC)=O)CN(C(=O)COC2CCCOC2)CCC12CCC2 c1(C(N2C(C)CCC(NC(C3CC4(CSC4)C3)=O)C2)=O)cnc2cccnc2c1 C1(CNC(CSC)=O)CCC(NC(=O)CCC(=O)Nc2nccs2)CC1 c1(C(=O)NCC(N(C(=O)C(C)OCC)C(C)(C)CC)C2CC2)cncc(CO)c1 C(c1ccccc1)=CC(=O)NC1CC(C(N2CCCC(CCCO)C2)=O)C1 Cc1c(C(=O)NCC2CCCN(C(=O)CC3CCC(C)(C)C3)C2)ncn1C C1(C(=O)NCC(CNC(C(CC(=C)C)OC)=O)(C)OC)Cc2ccccc2S1 C1(NC(=O)NCCCNc2ncc(C3CC3)s2)CC2CCCCN2C1 c1(OC)sccc1C(=O)NC(C)CN(C)C(c1ncn(C(C)C)n1)=O N1(CCCCOC)CCC(C(=O)NCC(O)CCC(=O)O)C(C)(C)C1 c1(OC)ccc(SCCC(=O)NC2COCC2NC(C2CSC2)=O)cc1 c1(C(=O)NC(c2occ(C(=O)NCc3c(C)ccnc3)n2)C)cc(C)nc(O)c1 C(=O)(CCCC(=O)NCCCCC(=O)NCc1ncc[nH]1)OCC C1(NC(C2C(C(=O)OC)CC2)=O)CCCN(C(=O)Nc2ccc(C(C)(C)C)[nH]2)C1 C#CCC(CC#C)C(=O)N1CCCC(CCNC(=O)C(C)Oc2cccnc2)C1 CS(=O)(=O)c1cc(C(N2CC3CC2(CNC(=O)COC2CCCOC2)C3)=O)co1 c1(OC)cncc(C(=O)NCCC2CCCN2C(=O)COCC2CCOC2)c1 c1(C(N2CCC(N(C)C(c3cnsn3)=O)C2)=O)cc(Br)cc(F)c1F c1(C(N2C(CNC(CCCNC(C)=O)=O)CCCC2)=O)cc2nc[nH]c2cc1N C1(NC(Cc2cccc(C)c2)=O)CC2CN(C(C3(O)CCCC3)=O)CC2C1 C1(CC(=O)NCC(CC)C)CN(C(c2cc(OC)cnn2)=O)C(C)(C)C1 CC1(O)CCCCC1NC(=O)C(F)CC1CN(C(C2CCCC2F)=O)C1 C(=O)(C1CCCc2scnc21)NCCC(CNC(C1CC2(CC2)C1)=O)O c1(OC)ccc(C(=O)NC2(CCNC(C3(O)CCCCC3)=O)CCC2)cc1 CC1(C)CCCOC1C(=O)NCC(c1ccccc1)NC(=O)C1=C(Cl)CCC1 C(=O)(C1=CCC(F)(F)CC1)NCC=CCNC(C(CO)NC(C)=O)=O c1(C(=O)NCCC(C)NC(=O)C(c2cccc(F)c2)F)cccn(C)c1=O C(C)(CNC(=O)CC1CCCN1C(C)=O)(C(C)C)NC(c1cnc(CC)s1)=O C(=O)(C(CC(C)C)C(C)C)NC1C(CC(N(OCC)CC)=O)CCCC1 C1(CN(C(=O)CC23CCCC2C3)CC)CCN(C(c2cc(OC)n[nH]2)=O)CC1 C(=O)(C(O)Cc1cnc[nH]1)NC(CN(C(CCC)=O)C)CC N1(C(C2CCC3(CC3)C2)=O)CC2CCN(C(=O)C(F)(F)CO)CC12 c1(CNC(C2(C(C)(C)O)CC2)=O)cccnc1C.CC1(C)C(C(=O)NC)C1C(F)F CC1(C)CC(NC(=O)C(C)(F)C(C)(C)F)CN(C(c2ccccc2)=O)C1 c1(C(=O)NC2CN(C(C(C)C3CCCC3)=O)CC(F)C2)cnc2[nH]cnc2c1 N1(C(Cc2c(C)scc2)=O)CC(NC(C2(C3CCCCO3)CC2)=O)CC12CCC2 C1(C(=O)NCCOCCN(C(=O)CN2CC3CCC2C3)C)CCC(O)CN1C.C=O Cn1[nH]c(C2CCCCC2NC(=O)NCC(CNC2CC2)C(=O)O)nc1=O C(C)(CCCN=c1ccnc(-c2ccc(OC)cc2)[nH]1)NC(CC=C)(C)C C1(N(C(C2CCCN2C)=O)CC2C(c3ncc(C)o3)C2)CN(C(C)C)CCC1O c1(OC)cccc(C(=O)NCCOC(F)F)c1NC(c1ccc(NC)c(F)c1)=O C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)C(C)(C)n2cccn2)CC1F C1(CNC(C(CC=C)NC(C)=O)=O)CC2CCC1N(C(c1cc(Cl)no1)=O)C2 Cn1oc(C(N2CCCC(NC(c3ccc(-n4cccc4)nc3)=O)C2)=O)cc1=O C(CCCC(=O)N1CCCC1C1(NC(=O)C(c2ccccc2C)C)CC1)(OC)OC c1(C(=O)NC(CC)CNC(C2CC3CCCC(C2)C3)=O)ccc(F)cc1[N+](=O)[O-] N1(C(C2C(CCC)C2)=O)CC2CCC2(CNC(c2cnc(S)n2C2CC2)=O)C1 N1(C(C2CC(=C)C2)=O)CC2CCC(Nc3nccc(COC)n3)C2C1 C(=O)(C1COc2ccc(Cl)cc21)NCCC1CCCN(C(CSC)=O)C1 c1(C(N2CCC(NCc3ccc(C)c(F)c3)C2)=O)c[nH]c2cc(C#N)ccc12 CCCCC(C)(F)C(=O)N1CCOCC(CNC(C2(COC)CCCC2)=O)C1 C1(C#N)(C(=O)NCC(CC)(CC)NC(=O)C(C2CCCC2)OC)CCC(=O)CC1 c1(C(=O)NC(CNC(C(CCC)CC)=O)(C)CO)ccc(S(=O)(=O)N(C)C)o1 N1(Cc2nnc(C)s2)CCC2(CC1)CN(C(c1ncn(C(C)C)n1)=O)CC(C)O2 C12(NC(C=CCN(CC)CC)=O)CCC(CC1)N(C(=O)C(CCSC)OC)C2 CCCCCC(F)C(=O)NCC(O)CNC(c1ccc(CNS(C)(=O)=O)o1)=O C(C(C)(COC)CC)NC(C(C)N(C(CCC)=O)C)=O Cc1nc(=NCC2C(C)CCCN2C(=O)Cc2ccc(F)cc2F)c(C#N)c[nH]1 C1(NC(C(COC(C)=O)O)=O)CN(C(=O)C=CC(C)(C)SC)CC1n1cccn1 N1(C(CCOCC)=O)CC(CNC(=O)CSc2n[nH]c(C)n2)C2(CC2)C1 N1(C(c2ccc(C)cn2)=O)Cc2ccccc2C(NC(C2(CF)CCC2)=O)C1 C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(=O)CC(C)P(C)(C)=O)C2(CCOCC2)C1 CC1=C(C(=O)NC2CC(C(N3CC(C(N)=O)C(C)C3)=O)C2)CCC1 O=C1CCN(CC(N2CCC2C2CC(F)(F)C2)=O)C(=O)O1 C1(CNC(=O)Cc2cscc2Br)CCC2(CCC2)C1NC(=O)C1CC1 Cc1ccc(C(=O)NCC(CC(C)C)NC(=O)C(c2ccc(Cl)cn2)(F)F)cn1 c1(C(=O)NC2(CNC(C3N(N=O)CCC3)=O)CCC2)cc2n(n1)CCCN2 C(=O)(CCCCCC#N)N1CCCC(C)(CNC(c2oc(CC)c(C)c2)=O)C1 c1(CNC(c2cc(C(=O)OC)[nH]c2)=O)cc(O)nc(CNC(=O)CCC2CC2)n1 C(CCC(C)(F)F)C(N1CCC(C2N(C(CCC3CC(C)C3)=O)CCC2)C1)=O CC1(C)CN(CC2=NC(=O)C=CCCC2)CCC1NC(=O)C1=CCCC1 n1(CC(=O)NC(CN(C(c2cnns2)=O)CC)C)nccc1C N1(C(c2nc(C)oc2)=O)CCN(C(c2cc(Cl)ns2)=O)CC1c1nccn1C N1(C(C(C(C)C)O)=O)CCCC2(C1)CN(C(c1ccnn1CCF)=O)C2 C(=O)(C1CCOc2c(F)cccc21)NCC(CNC(Cc1cc(CC)no1)=O)O Oc1ccc2c(c1)CN(c1nc(NCC(Cl)Cl)nc3c1ncn3C(F)F)CCO2 c1(C(=O)NCCCC(CCC)NC(C(CC=C)C)=O)noc2ccccc12 c1(C(=O)NC2CN(C(c3c(SC)cccn3)=O)C(C)(C)C2)cc(F)c(F)c(F)c1F N1(C(C=CCOC)=O)CC2CCN(C(c3cnc(C(C)C)nc3C)=O)CC(C2)C1 C1(NC(C2N(CC(C)C)CCC2)=O)CN(C(=O)C(C)OC2COC2)CC1C N1(C(C(=O)NC(CCC)C)=O)CCn2c(nc(OC)c2Br)C1 C(=O)(CC(C)(C)C(C)=O)NC(CCC)C(N1CCCCC(N2CCC2)C1)=O C12(C(=O)NC(CC)C3CCC3)CC3CC1C2C3.C12CCC1CNC2=O C1(NC(C(c2n(C)ccc2)=O)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC2C1 CCC(C)(C)C(O)C(=O)NC1CCN(C(=O)Cc2ccc(S(=O)(=O)NC)s2)C1C N1(C(c2c(C)onc2)=O)C2CCC1C(F)C(NC(=O)CCn1ncn(C)c1=O)C2 O=C(C(c1cn[nH]c1)=Cc1ccc(F)cc1)OC1CC2C(C1)C2(F)F C1(CNC(C=C=C(C)C)=O)CCN(C(=O)CCCC2CCC2)CC1(F)F C1(C(=O)NCCOC(CNC(CCc2nc(C)sc2)=O)(C)C)OCCOC1C CC1(C)CN(C(C2(CO)CCCO2)=O)CC(CNC(c2coc(CO)c2)=O)O1 C1(C(=O)NC(=O)CN2CCC(C(=O)NCC3CC3)CC2)CC2CCCC(C1)C2 CC1CC(NC(c2cc(-c3ccccc3)oc2Cl)=O)CN1C(c1ccns1)=O CN1CCC(C#N)(C(=O)NCCC(O)CNC(C2CCn3cncc3C2)=O)CC1 C12(CNC(c3cnc(COC)s3)=O)CCC(Nc3nccc(C#N)n3)(CC1)CO2 C1(CNC(C(C)=O)=O)CN(C(=O)CC(c2ccc(F)cc2)O)CCCO1 N1(C(CCNC(c2nc(C)sc2)=O)=O)CC(C(=O)NCC(C)C)C(F)C1 C(C(CC1CCCC1)C(=O)NCC(C)SCC(F)F)NC(C(=O)NCC)=O c1(OC)cccc(-n2nc(-c3cncs3)nc2-c2cnn(CC3CC3)c2SC)c1 N1(C(Cn2c(C)ncc2)=O)CCC(C2(NC(=O)C(C)S(C)(=O)=O)CC2)CC1 Cc1cc(C)n(CC(=O)NCC2CN(C(=O)C(O)c3cnc[nH]3)CC2O)n1 c1(C(=O)NC2CC(NC(c3c(C(=O)OCC)scc3)=O)C2)nncc2c1CCCC2 N1(C(C(n2c(C)ccn2)C)=O)CCCC(C2CN(C(=O)C3=CCCOCC3)C2)C1 c1(C(=O)NCCC2CC(NC(=O)CC3(n4ccnn4)CC3)C2)cc(Cl)c[nH]1 c1(C(=O)NCc2c(CCNC(CC(COC)C)=O)ocn2)cc(C)c(Cl)cc1F c1(C(=O)NC2C(CNC(C(CCOC)C)=O)CC2)ccc2c(c1)C(=O)NCC2 C1(C(N2CCC(OC(C)=O)C2)=O)CCC2CCC1N2C(=O)C(F)n1ccnc1 NS(=O)(=O)CCCC(=O)NCC(CO)NC(=O)CSCc1ccncc1 CCC(C)C(C(=O)N1CC(C)(C)CC1C(=O)OC1CCCCC1)NC(C)=O C1(C(=O)NC2C(NC(c3c(OC)ncc(F)c3)=O)C2)CCC2CCC(=O)N2C1 Cc1scc(C(=O)NCC(C(=O)NCCc2ncon2)N(C)C)c1C c1(OC)cnc(Cl)cc1C(N1CCOC(CNC(=O)CC2CCCOC2)C1)=O N1(C(c2cnc(C(C)(C)CF)o2)=O)CCCC2C(NC(=O)C(N)=O)C(C)(C)C12 N1(CC)CC2(C(=O)NC)CC1C2.C1(C(=O)OC)COC(C)C1 CCC(C)(CO)C(=O)NCC1(CNC(c2ccc[n+]([O-])c2)=O)CCCCC1 C1(N(C(C2N(CC)CC2)=O)C)CCN(C(c2cscc2OC)=O)CC12CC2 C#CC1(NC(=O)Cc2cc(C(=O)OCC)cs2)CCCC(C)(C)C1 CC(CC(C)(C)C)C(=O)NCC1CC1CNC(c1cc(C2CCC2)nn1C)=O N1(C(C(CC)N(C)C)=O)CC2(NC(=O)CSCc3cc(C)ccn3)CC1C2 CCCC(CNC(=O)CC=Cc1cccnc1)C(=O)NOCCCOCC C123CC1CN(C2)C3=O.c1(C(C)NC(c2nc(Br)cs2)=O)cccc(Br)c1 N1(C(=O)NCC(c2cccc(Cl)c2)C)CCSC2COCCC12 C(=O)(C#CC1CCOC1)N(CCNC(C1(CCc2ccccc2)CC1)=O)CC c1(C(=O)NCC2C(NC(C(Br)=C(C)C)=O)CCC2)cc2c(nc1N)CCC2 c1(C(N2CC(CCNC(C(CC)C(=O)OC)=O)C2)=O)ccc(Cl)c2ncccc12 c1(C(N(CC(=O)NCC(n2cccn2)C)CCC)=O)cnncc1NC c1(NC(C2(NC(C(C)=CCC)=O)CC2(C)C)=O)ccc[n+]([O-])c1 c1(C(=O)NCCc2cnc(NC(=O)Cc3ccccc3F)s2)cc(Cl)nc(Cl)c1Cl C#Cc1cccc(C(=O)NCC2CC3CC3N2C(=O)CCc2cscn2)c1 C1(C(N2CC(NC(c3c(C)nc[nH]3)=O)C(O)C2)=O)CCC(C)(O)CC1 c1(OC)cccc2c1OCC(C(=O)NCCCc1cn(C3CCOC3)nn1)C2 C1(C(=O)NCC(CC)NC(C2CC(OC)C(OC)C2)=O)(CF)CC2(CCC2)C1 N1(C(C(C)Nc2scc(C)n2)=O)CCC(CNC(c2nccs2)=O)C(C)C1 N1(CC(=O)N(CC(C)NC(=O)CSc2cccc(O)c2)C)CCS(=O)(=O)CC1 N1(C(c2c(SC)ccs2)=O)CC2CCC1C(CNC(=O)CN1CCN(C)CC1)C2 CC1(C)CC(CC(N2CCC3C(NC(=O)CN4CC=CC4)C3C2)=O)CCO1 N1(C(c2cnc(O)o2)=O)CC2CCCC(C1)N2C(=O)C(CO)C(F)(F)F N1(C(=O)Cc2ccsc2)CCC2CCN(C(c3ccncc3O)=O)CC2C1 C(CCCC(CO)NC(C1CC2(C1)CC2F)=O)NC(c1c(C)nn(C)c1)=O c1(CC)ccc(C)c(C(N2CC3CC3(NC(=O)CN(C)CCO)C2)=O)c1 c1(C(=O)NC(C)CCCNC(=O)Cc2cncs2)ccc2nc(CO)[nH]c2c1 N1(C(C(CC)C(C)C)=O)CCCC2(CCN(C(c3ccnn3COC)=O)C2)C1 N1(C(C2CC(C(C)=O)C2(C)C)=O)CCOCC(CNC(=O)CN2CCCC2=O)C1 N1(C(C(F)OC)=O)CC(NC(C2(C)CNC(=O)C2)=O)CC2(CC2)C1 C12(C(N(C3CCCC3)CCCC)=O)CCC1CN(C(c1c(C)nsc1N)=O)C2 C(=O)(C1CCc2ccccc21)NC1C(C)CN(C(=O)CC(N(C)C)C2CC2)C1 c1(C(=O)NC2CCN(C(C=Cc3c(C)cncc3)=O)CC2)cc(S(N)(=O)=O)cs1 C1(OCC)(CNC(=O)CC2CCCC2)CN(C(C2CC2Cl)=O)C1 c1(OC)cc(C(=O)NC(C2CCCN2C(c2cn3c(n2)SCC3)=O)C)cc(C)c1 N1(C(C(C(C)C)OCC)=O)CC(C)(C)CC1CC(N1CCCN(C)CC1)=O C1(C(=O)N(C2(C)CCN(C(CN(c3ccccc3)C)=O)C2)C)CC2(CCC2)CO1 Cc1ccc(F)c(CN2CC(C)CC2C(=O)Nc2ccc(Cl)c(Br)c2)c1 CCCCCCC(CC)C(=O)NCC1(NC(=O)C(F)C(F)(F)F)CCCCC1 CC1(CC(=O)NCC2CCOC2C(N2CCC(C(F)F)C2)=O)CCOC1 N1(C(C2CC3(CC3)C2)=O)CC(C2CC2)(C(N2CC3CC3C3CC23)=O)C1 n1(CC(=O)NC2C(NC(=O)COCc3ccncc3)C2)ccccc1=O C(C(C)(O)CNC(=O)CC1(C2CC2)CC1)NC(CN(C1CC1)CC)=O CC1CC(C(N2CCOCC2CN(C(=O)C=CC(N)=O)C)=O)CCO1 C12(C(N(C)Cc3c(CNC(C(C)OCC)=O)cccc3)=O)CCCN1CCC2 c1(C(=O)NCC2(C)CCC(NC(=O)CCc3cnn[nH]3)C2)cn2ccsc2n1 C1(C(=O)NC(C(=O)OCCC)C)OCCC1CNC(=O)CSCCF c1(Oc2cc(-c3cn(COC)nc3)ncc2)cccc2c[nH]nc12 CC1(C)CCC(CO)(NCC(=O)Nc2ccc(CN)c(F)c2)C1 c1(NC(N2C(C)c3cccn3CC2)=O)ccc2c(c1)NC(=O)C1CCCCN21 c1(C(N2CCC(CC(=O)NC(c3nc[nH]n3)C)C2)=O)cnn(C(C)(C)C)c1N Nc1c(C(N2CC(NC(C3C4CC5C(C4)C35)=O)CC(F)C2)=O)ccc(Cl)c1Cl C1(C(=O)NC(CC=C)CC)CCN(C(C2CC(C(C)C)C2)=O)C12CCC2 c1(C(=O)NC(C2CCN(C(=O)C(C)(C)CN(C)C)CC2)C)ncc2[nH]ncc2n1 C1(C(=O)NC2CC(C)(C)N(C(c3cccc[n+]3[O-])=O)C2)CCCC2(CCC2)O1 Cc1scc(C(=O)NCCC2CCCN2C(C2(C)CC2C)=O)c1Br S(=O)(=O)(c1ccc(C(=O)OC)cc1)N1CC2CN(N(CCC#N)CC)CC2C1 Cc1ccc(CC(=O)NC(C)(CNC(C2CCC2(C)C)=O)CO)s1 C1(C(N2CCC(CC(N3C4(C)CC4CC3)=O)C2)=O)CC2(CCCO2)C1 C1(NC(c2c(C)ccs2)=O)CCN(C(c2cc(-c3cnn(C)c3)no2)=O)CC1O C(C(C)(C)CN(C)C(c1ccc(CO)o1)=O)NC(CC=CCC)=O C1(NC(c2nnn(CC)c2C)=O)CCN(c2nc(Cl)ncc2C)CCC1CO c1(C(=O)O)cnn(CC)c1CC(C)C.C(c1cnc[nH]1)=CCN(C(C)C)CC c1(OC)ccccc1NC(=O)C(c1ccc(C(N)=O)s1)N1CCC(CN=[N+]=[N-])C1 C1(NC(=O)C2=CCC2)CC2CCC(C1)N2C(=O)Cc1nc(C2CC2)cs1 N1(CCC(=O)N(C)CCNC(=O)CCSc2ccc(F)cc2)CCN(C)CC1 Cc1c(NCC2CCCCS2(=O)=O)nc[nH]c1=NCC1CCCCC1(C)C C1(C(N(CC(CNC(c2c(OC)nccc2)=O)O)C)=O)CCCN1S(=N)(=O)N(C)C C1(C(N2CCC(C(=O)NC)C2C)=O)CN(C(c2ccccc2F)=O)CC12CCC2 C1(C(N(C)C)=O)CC(F)(F)CN1C(c1cccc(N(C)C)c1)=O c1(C(N2CC(CNC(C(C)C)=O)C3(C2)CC3)=O)cc(F)c(Cl)cc1Cl C(=O)(C1=C(Cl)CCCC1)NCC1(F)CCC(CNC(C(=O)N(C)C)=O)CC1 C1(C)(C(N2CCCC(CCC(=O)NC(CC)COC)C2)=O)CCC2CC2C1 N1(C(C(Cc2c(C)nn(C)c2C)C)=O)CCCN(C(=O)CCCCC(F)F)C(C)C1 C12(C(N3CCOCC3)C(=O)NCCCF)CC(CO1)N(C(=O)C1=CCOCC1)C2 C(N=c1cc(C#N)nc(C2CC2)[nH]1)C1(NC(C2CCCC(C)C2)=O)COC1 Cc1ccc(CN2CC3(CN(C(c4cn(C)cn4)=O)C3)C2)cc1I Cc1ccc(C2(NC3CC(NC(=O)Nc4nc(O)sc4C)C3)CC2(F)F)c(C)c1 N1(C(C)=O)CC(C)CN(Cc2cccc(C(F)F)c2C)CC1C C1(NC(=O)CCn2cccn2)C2COCC1CN(C(=O)CCN1CCOCC1)C2 N1(C(c2n(CC)cc(Cl)c2)=O)CCN(C)C(CNC(c2ccc(C)c(F)c2)=O)C1 C(=O)(C(O)C1=CCCCC1)N1C(C(=O)NC2CC2O)C2CCC1C2 Cc1cncc(C(=O)NC(Cn2ccnn2)C(=O)NC2CC(CCF)C2)c1 CC(C)C(CC(=O)N1CC(C)=C(C)C1)NC(c1nc[nH]n1)=O CC(C)(C#N)C(=O)NC1CCN(C(c2cnc(-c3ncccn3)s2)=O)C1 CC(N=c1[nH]c2c(c(=NCCCCC#N)[nH]1)SCC2)N1CCc2sccc2C1 Cc1c(C(=O)NCC2CCN2C(=O)CCCCC(F)(F)F)oc2c1C(=O)CCC2 C#Cc1ccc(Cl)c(C(=O)NCC2(F)CCN(C(=O)C(CCOC)OC)C2)c1 CC1N(C(C2CC(O)CN2C(C2CC(F)CN2C)=O)=O)CC(C)OC1(C)C N1(C(CCOCCC)=O)CCC(NC(C2CCCS2)=O)C(C)C1 C(=O)(CCCOC1(Cc2ccccc2)CC1)NC1(CNC(C(C)=CC)=O)CCC1 C1(C(C)NC(c2ccc(F)o2)=O)CCN(C(=O)C(C)C(C)O)CC1 c1(C(=O)NC2CCN(C(c3nnc(C)s3)=O)CC2C)c(F)ccc(F)c1F N1(C(C(C)(c2ccccc2)OC)=O)CC2CC(NC(c3coc(Br)n3)=O)C2C1 C#Cc1ccc(C(=O)NC2(CCNC(C3CCCCC3F)=O)CCC2)c(OC)c1 C1(NC(C2(O)CCC2)=O)CC2(C1)CC21CC1.C1(C2C(=O)N2)(C(C)C#N)CCCC1 C1(CC)CN(C(c2cc(C)sn2)=O)CCN1C(C1CCC1(F)F)=O C1(C(N2CCC(CN(C(C(C)NC(C)=O)=O)C)C2)=O)CCc2cnn(C)c2C1 c1(C(N2CC(CCCNC(C(C)N(C)C)=O)OCC2)=O)c(O)cccc1F S(=O)(=O)(c1cccc(C(=O)NCCCCCCNC(c2conc2C)=O)c1)NC C#CC1(C(=O)NCc2noc(C(C)O)n2)CCN(C(=O)OC(C)(C)C)C1 N1(C(CN2CCN(CC)C(=O)C2=O)=O)CC2CC1CN(C(C1CC1C(N)=O)=O)C2 C1(c2n(CC=C)nnn2)(NCCCn2cccn2)CCC2C3CCC123 N1(C(CCCOCC)=O)CC(NC(c2conc2C(F)(F)F)=O)CC12CCCC2 C(=O)(C(C)(O)C(C)C)N(CCNc1c(NC(=O)C(=O)N(C)C)cccc1)CC CC1(C)C(CNC(c2cc(Cl)sc2Cl)=O)CCN1C(=O)C=Cc1nccs1 CON(CCC(=O)N1CC=CC(OC)C1)C(=O)C1CCN(C)C1 c1(C(N2CCN(C(CS(CC)=O)=O)C(CF)C2)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-] C(=O)(C(C)C1=CCCC1)NC1(CC=C)CN(C(c2ccn(C)c2C)=O)C1 C(=O)(C1=C(F)CN(C(=O)CC2CC2CCC)CC1)NCCCC(=C)C Cc1ccc2ncc(C(=O)NCC(C)CNC(=O)CC3CC3C3CC3)n2c1 C(=O)(C(CC(F)F)N(C(=O)C(C)c1ccco1)C)N(C(C)CCO)C N1(C(C(CC)OC)=O)CC(CNC(=O)Cc2cc(F)ccc2OC)CC(C)C1 c1(C(=O)NCC2N(S(C(C)C)(=O)=O)CCCC2)c(Br)ccnc1Cl N1(C(C(C2CCC(C)CC2)CC)=O)CCCC2CN(Cc3cc(OC)n[nH]3)CC12 C1(NC(C(COC)C)=O)CCCCC12CCN(C(C1CSCCS1)=O)CC2 C1(NC(c2scc(CNC(c3scc(C#N)c3)=O)c2)=O)CN2CCC1(F)CC2 N1(Cc2cc(OC)c(O)c(I)c2)CC2(CCN(C(=O)C(C)(O)C(F)(F)F)CC2)C1 C1(C(=O)NCC(C)N(C(=O)CNC(c2ccccc2O)=O)C)CC12CC(C)(C)C2 C(S(=O)(=O)c1ccc(Cl)c(Cl)c1)c1ccc(NC(C=CCC)=O)cc1 C1(C(=O)NCC=CCNC(=O)COC(C)CC)(C(=O)OC)CCOCC1 C1(C#N)(COC)CN(C(=O)CCC2CCC(NC(=O)C(F)OC(F)(F)F)C2)C1 CC1(CNC(c2ccsc2)=O)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1 CCCCC(C)CCC(=O)N1CCCCC1CCN(C(=O)CCCCCSC)C N1(C(CCCC2(C)N=N2)=O)CC2C(C(=O)Nc3ccc(C(=O)N(C)C)cc3)C2C1 N1(C(C(C)OCCC(C)C)=O)CCC(C)C(CNC(c2cc(C#N)n(C)n2)=O)C1 C1(CC(=O)NCC2N(C(c3cc(-c4cn(C)nc4)[nH]n3)=O)CCC2)CC2COCC12 N1(C(c2cccnc2)CC)CCOC(O)CC1 C(=O)(CCCC(N)=O)NC1C(NC(C2CCCN(S(CC)(=O)=O)C2)=O)C1 C12(NC(c3cn(C)nn3)=O)CCC1CN(C(=O)C(O)Cc1cccc(Cl)c1)C2 C(F)(C(=O)NNc1c(F)c(F)cc(F)c1F)n1cc(CC(=O)OC)nn1 c1(NC(C2N(Cc3c(OC)cccc3)CCC2O)=O)ccc(Br)cc1C(N)=O C1(C)(NC(CCNC(COC)=O)=O)CCCCC1C(N1CCCCC1C)=O N1(C(c2scc(C#N)c2)=O)CC2OCC(NC(=O)CCn3cncn3)C2C1 c1(C(N2C(C)CN(C(=O)C3=CCCC3C)CCC2)=O)ccc2c(ccn2C)c1 O=C1CCCC2C(C(=O)NOCC(N3CCCC(F)CC3)=O)C12 C1(NC(C2N(CC)CC2)=O)CN(C(c2coc(OCC(F)(F)F)n2)=O)CC1(C)C C1(C(N2CC(F)(C(=O)NCC3(F)CC3)C2)=O)CCNC1=O N1(C(CSCCC)=O)CCCC(N(C)C(c2ccccc2SC(C)(C)C)=O)C1 C1(Nc2c(C#N)cncc2)CC2CN(C(C3C4COCC34)=O)CC2C1 CC(CBr)N=c1cccc(S(=O)(=O)NC2CC(CS(C)(=O)=O)C2)[nH]1 C#Cc1ccc(C(N2CCCC(C)(C)C2CNC(c2ccoc2Cl)=O)=O)cc1F Cc1cc(C)n(C(C)C(N2CCC(C(C)C(N3CCC(C(F)F)C3)=O)CC2)=O)n1 c1(NC(C(CNC(CCNC(COC)=O)=O)CC2CCCC2)=O)cnc(Cl)c(C)c1 c1(CC)ccc(Cl)c(C(N2CCC(N(C(=O)Cc3nncn3C)CC)C2)=O)c1 c1(-c2onc(C(c3ccccc3)CN(C)C)n2)ccc([N+](=O)[O-])cn1 CCCCC(=O)C(=O)N1CC(OC2CCN(C(c3ccoc3)=O)CC2)C1 N1(C(C2C(C(=O)OC)C2(C)C)=O)CC2CC2(NC(=O)Cc2scnc2C)C1 c1(C(=O)NCCC(=C)CNC(=O)C=Cc2scnc2C)cc(Cl)c2c(c1)OCO2 C(C(CC(C)C)C(=O)OC)c1c(OCC)c(F)ccc1.c12ocnc1C(=O)OC2 CC1=C(C(=O)NCCCC(C)NC(C2CC3C(C2)C3(F)F)=O)SCCO1 c1(C(=O)NCCNC(c2nn(C)c3c2CCC3)=O)ccc2c(c1)CCC2(F)F CCCC(C)C(=O)NC1CN(C(c2cnn(C(C)C)c2C)=O)CC1CC N1(c2nc(C)nc(Cl)c2)CC(NC(C2OC(C)CC2C)=O)C2(CCOCC2)C1 c1(C(N(C2CCN(C(C3CC(=O)N(C4CC4)C3)=O)C2)C)=O)cn2ncccc2n1 N1(C(C=CCCC)=O)CCC(N=c2ccnc(CC)[nH]2)C(C)C1 C1(NC(Cc2c(C)noc2C)=O)CN(C(c2ccnn2C)=O)CCC1C C1(N(C(C=C=C(C)C)=O)C)CCC2CN(C(=O)CCNC(=O)CO)CC12 c1(CC(C)NC(=O)C(=O)Nc2cccc(C(N)=O)n2)cccc(F)c1 c1(C(N2CC3(C(C(=O)NCCOCC#C)C3)C2)=O)cc(SC)ccc1Br N1(C(C2(C(C)C)CC2)=O)CCCC(C(=O)N(C2CCC(O)CC2)C)CC1 C(C(COC(c1cc(-c2cccnc2)nn1C(C)C)=O)C(C)C)OC c1(C(=O)NCC(C(C)C)NC(C(C=C)(C)O)=O)cnc2onc(C)c2c1 c1(C(=O)OC)cc2c(N(CC(C)NC(=O)CC3CC(C)(C)CO3)C)[nH]cnc-2n1 C(=O)(C(F)CC(C)(C)NC(=O)C(CO)C(F)(F)F)NCC(CC)CC(C)C C1(c2ccccn2)(Sc2n(C3C(c4cn(CC)nc4)OCC3)nnn2)CCOCC1 N1(C(c2ccc(OCC)nc2)=O)C2CCCC1CC(N(C)C)C2 C1(CC)CN(C)C(=O)CN1C(=O)CCCCCN(C)C(C1CC(=O)N(OC)C1)=O CCS(=O)CC(=O)NCCCN(C(c1cccc(-c2csc(C)n2)c1)=O)C1CC1 C1(C)(C(N(CCOC)C)=O)CC12CCN(CC13CCC(CC1)C3)CC2 Cn1ncc(C(=O)NC2CCCC2(C)C)c1F N1(C(CCCN(C(C)=O)C)=O)CCC(C)C(CNC(=O)CNc2cnn(C)c2)C1 c1(-n2cnc(CS(=O)(=O)NC(C(CC)O)=O)n2)ccc(C(C)(C)C)cc1 c1(CC)c(C(=O)NCC(O)CN(C(=O)C(C(C)C)c2ccccc2)C)csc1C C1(OCC)CC2(C1)CC2C(N1CCCC1C(C)NC(=O)CN1CCCCC1=O)=O c1(OC)ccc(C)cc1C(=O)NCC1CC(NC(=O)C=C2CN3CCC2CC3)C1 c1(OC)ccc(C(N2CCCC2CC(=O)NCC2C3CCCOC23)=O)nn1 CN1CCOc2cc(CN3CCOC(C(=O)Nc4cnn(C5CC5)c4)C3)ccc21 C1(C(C)NC(C2C(=C)CC2)=O)CCN(C(c2nn(C)cc2C)=O)C(C)C1 Cc1[nH]c(C)c(C(=O)NCC(CO)NC(c2cccc(CS(N)(=O)=O)c2)=O)c1C Cc1cc(C)n2nc(CC(=O)NC3(C)CCC(NC(=O)CSC4CC4)CC3)nc2n1 N1(C(C(CC)C)=O)CCC2(CC1)CC2NC(c1cc(F)ccc1C)=O C=C(Br)CCC(=O)NC(C1CCN(C(=O)C(C)n2ccnc2)CC1)(C)C C1(NC(C2(OC)CCSC2)=O)CCCCC1C(=O)NCCCP(C)(C)=O N1(C(C2C(C)C2(F)F)=O)CCC(C2CC2)(CNC(=O)CCn2ncn(C)c2=O)C1 C1(C(=O)NCC(c2ccccc2)F)COCCN(C(c2c[nH]cc2C2CC2)=O)C1 c1(CC2C(NC(=O)Nc3nc(C)nn3C)C2)c[nH]c2cccc(F)c12 N1(C(C(C)N(C)CCOCC)=O)CCCC(NC(=O)C(C)N(C)C)C1.C1CO1 CC1CN(C(=O)C(CC(F)F)NC(=O)C(C)N(C)C)CC1N=[N+]=[N-] C1(C(=O)NCC2(n3nccn3)CC2)(CC)CCCN1C(=O)CC1CC2CC2C1 c1(C(N2CC(CNC(C(CC)SC)=O)C(C)C2)=O)cc2nc(C)ccc2o1 CC1(C)OCCC1C(=O)NCC1CC(NC(=O)CNC(=O)C2CC2)CC1O N1(C(=O)CC2CCN2C(c2ccc(C(F)F)o2)=O)CC2CC3CC2C1C3 N1(C(c2cn(CCCC)nn2)=O)CC(NC(=O)C(CC)SC)C2CC2C1 Cc1noc(C)c1CCN(S(=O)(=O)CC1CCOC1)C Nc1cc(F)c(C(=O)NC2CC3CC(NC(C4CCC(F)(F)C4)=O)CC23)c(F)c1 Cc1ccc2occ(C(N3CCC4CCN(C(N)=O)CC34)=O)c2c1 c1(OC)ccc(F)c(CN2CC3CN(C(c4cc(F)ccc4F)=O)CC23)c1F c1(NC(C(N2CCC(C(=O)NCCC)C2)=O)=O)c(OCC)ccc2c1CCC2 C1(C(=O)NC2CCC3(CC3)C2)(CC)CCN(C(c2nccn2C)=O)CC1 N1(C(C)=O)CCCC1C(N1CC(O)(C(C)NC(=O)C(F)=CCCF)C1)=O c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)cnc(Br)c(N)n1 Cc1ccc(CCC(=O)N(CC(O)CN(C)C(C2(N(C)C)CC2)=O)C)o1 N1(C(C2N(C)CC2)=O)CC2CC(C1)CN(C(C1(C)CCCO1)=O)C2 c1(OC)cccc2[nH]c(=NCc3sccc3C)[nH]c(=NC(C)CN(C)C(C)C)c12 C=CC1(N(C)C)CCN(C(c2nc(Br)sc2C)C(=O)NCC(=C)C)CC1 N1(C(C2(C)CCCO2)=O)CC2(CO)CC1(C(N1CCNC(=O)CC1)=O)C2 c1(C(N2CC(C)CC(NC(C(C#C)(C)C)=O)C2)=O)ccc(F)c2c1CCC2 C1(C(C(=O)NCC(F)F)N(C2CC2)Cc2ccc(F)cc2)CCC2(CCC2)O1 C1(N(CC=C)CC2CCC2)(C(=O)NC(CC(N)=O)c2cn(CC)nn2)CCCCC1 C#Cc1ccc(C(=O)NC2C3CC(NC(=O)C(C)(CC)OC)CC23)cc1C Cc1ccc(OCCC(=O)NC2CC(Cn3cc(C4CCCC4O)nn3)C2)cc1 C1(CNC(C2CN(S(CC)(=O)=O)C2)=O)CN(C(c2cc(C)c[nH]2)=O)CC(C)(C)C1 c1(N2CCC(O)(C(C)NC(COC(CC)C)=O)C2)ncc2cccnc2n1 c1(C(C)N(C(CC2CCCC2)C(=O)NC2CCC2)C)cccc(F)c1 c1(CCNC(COCCC)=O)cnc(C)c(NC(=O)C(C)(COC)OC)c1 C1(C(N2C(NC(CONC(C3(C=C)CCC3)=O)=O)CCC2)=O)CC(C)(C)OC1(C)C Cc1cc(CC(=O)NC(=O)C(C)C(=O)O)ccc1-n1cccc1 CC(C)(C)C(C)(C)C(=O)NCC1CCN(C(C2CN(S(N)(=O)=O)C2)=O)C1 N1(C(c2coc(Cl)c2)=O)CC(NC(C23CC(O)C2C3)=O)CC12CCCC2 C1(C(N(C(CNC(Cc2nc(CC)sc2)=O)C)C)=O)CC(C)(C)CCO1 CCCC(CCNC(=O)C1=NOC(CNC(C2CCCCC2)=O)C1)CCC S(=O)(=O)(c1c[nH]ccc1=NCC1CCCOC1)N(C(c1ccc(Cl)cc1)C)C C1(CCNC(=O)CCOC2CCC2)CCN(c2nc(C3CCOCC3)ns2)C1 C1(CC(=O)NC2CCN(C(C3CC3C3CCCO3)=O)CC2)(CC)CCOCC1 Cc1oc(CNC(=O)CC2CNC(=O)O2)nc1C(N1CCCC1(C)C(C)(C)C)=O N1(C(C2(OC)CCCC2)=O)CCC(C)C(CNC(C2(F)CCCC2)=O)C1 C1(CCC)CCCN(C(=O)C=CC(C)NC(=O)C(C)CC2CC2)C1 c1(OC)cc(OC)c(C(N2CCN(C(=O)Cc3ccsc3)C(C(C)C)C2)=O)cn1 c1(OC)ccc(C(=O)N)c(C)c1.N12CC3(CCC1C3)NC2=O.C(C(C)(C)SC)=C C=CC(CCC)CC(=O)N1CCC(C)(NC(=O)CC2C=CCC2)CC1 C(=O)(CCC(=O)N1CCC(C)(CCNC(=O)CCNC(=O)CCC(C)C)C1)OC C1(C(=O)NCC(CC)(CC)NC(=O)C#CC(C)(C)O)CCc2cncn2C1 c1(COCCOC)ccc(C(=O)NCC(C)N(C)C(C2(O)CCSC2)=O)cc1 C(CC(=O)Nn1ccnn1)(C(C)(C)C)NC(c1c(C)cc(C)cn1)=O c1(C(N2C(C#N)CC2)=O)cc(-c2cc(F)ncc2F)c2[nH]ccc2c1 c1(-c2nc(C)sc2)cccc(CNC(=O)C(=O)NCCC(O)C(=O)O)c1 C(CCC(O)C(=O)NCC1(CO)CCOC1)NC(C1(OC)CCCCC1)=O N1(C(c2c(C)ccc(C)n2)=O)CCN(C(=O)Cn2cnnn2)C(C)C1C N1(C(C2(C)CCOC2)=O)CC2CN(C(c3ccc(N4CCOCC4)nc3)=O)C2C1 c1(C(c2cn(CCOC3CCN(C(=O)CCF)C3)nn2)O)ccccc1Br CC1CCC=C1C(=O)N1CC(NC(c2ccc(OCF)cc2)=O)C2(CC2)C1 Cc1cc(C(N2CCC(C)N(C(c3nnsc3N)=O)CC2)=O)c(C)c(C)c1 N1(CCC(=O)NCC(CNC(c2c(CC)nccn2)=O)(C)O)CCP(C)(=O)CC1 c1(CC)cc(C(N2CCOCC(NC(c3csc4cncn34)=O)C2)=O)cc(O)n1 N1(C(C23CC(OC)C2C3)=O)CCC(CNC(=O)CCc2csc(C)n2)CC1C C1(C2(NC(CC=C(C)C)=O)CC2)CCCCN1C(C1CC2CC2C1)=O c1(CCNC(C=CC(C)NC(=O)C=CC(C)(C)C)=O)noc(=O)n1C c1(CC(=O)NC2C(NC(CC(=O)OC)=O)CCOC2)c(F)c(F)c(F)c(F)c1F c1(C(N2CCCCC2c2cn(CC3CC3)nn2)=O)ccc2c(c1)OCCCO2 C(=O)(CCCC(=O)NCC)N1CC(CNC(COCC(=C)C)=O)C(C)C1 c1(C(=O)NC(C2(O)CCN(C(=O)C3=CSCCO3)C2)C)cc(F)c(CO)c(F)c1 c1(C(=O)NCC(CNC(C2(OC)CCCOC2)=O)O)cc2ccccc2nc1O Cc1nc(N(C2CN(C(=O)C=Cc3c(F)cccc3F)C2)C)cc(C#N)n1 N#Cc1c[nH]c2ncnc(N3CC4CCN(C(c5ncc(Cl)cc5Cl)=O)C4C3)c12 C(=O)(C(CC)CC(C)C)NCC1N(C(c2c(CC)nn[nH]2)=O)CCCC1 N1(C(c2ccn(CC(C)C)n2)=O)CCC2(NC(=O)C=Cc3ccsc3)CCCC12 N1(C(Cn2c(C)nc(C)n2)=O)CC(NC(=O)CC2CCCNC(=O)C2)CCC1C N1(C(c2c(CC)cccc2)=O)CC(C)(C)CC1CNC(C1CCCO1)=O C(=O)(CC(C)(C)C(=O)N(CC(C)CNC(c1ccc(F)s1)=O)C)OC C12(C(=O)NCCOCCNC(c3c(OC)csc3)=O)CCCC1(C(N)=O)C2 C=CCC(CNC(C1CSCCN1C(=O)C=C(C1CC1)C1CC1)=O)CC(C)C c12ccc(Cl)c(c1)C(=O)N1CC(C1)C(F)C(=O)N2.c1(OCC)cccnc1OC Cc1ccc2nsnc2c1C(=O)NC1CCN(C(=O)C=C2CCCCC2)CC1F c1(C(=O)NC(C2(O)CCN(C(c3c(CC)scc3)=O)C2)C)cc([N+](=O)[O-])c[nH]1 c1(NC2(C)CCC2)ccnc(Br)c1F.C12(CC1)N(C)C(=O)NC2 n1(CC=C)nnnc1C(c1ccn(C)n1)NCC1CC1 C(C(C)C(=O)NCc1ccc(C(=O)NC(c2nc(C)cs2)C)s1)SC c1(C(=O)NC2(CNC(c3cc(Cl)no3)=O)CC3CCC2C3)ccnc2ncnn12 n1(CCC)cc(C(c2nnnn2C2CC(F)(F)C2)NCC(C)(C)OC)nn1 C1(CNC(C2(CC#C)CCCCO2)=O)(CO)CCN(C(C2(O)COC2)=O)CC1 Cn1cnc(C(N2C(C(=O)NCC3CC(C)(C)C3)CCC2C2CC2)=O)cc1=O c1(CC)c[nH]c2cccnc12.C12C(CC)CCN1C(=O)CC1CCCC1NC2=O Cc1cccc(C)c1CC(=O)NC1CCC(CCNC(=O)C(Cl)=CCl)C1 CC1OCCCC1C(=O)N(C)CCOCCN(C(=O)Cc1cccnc1)C C(C1=CCCCC1)NC(c1n(CCCCCC)nnn1)(COC)C1CC1 c1(C(=O)NCCOCCNC(C2COC(=O)O2)=O)cccnc1-n1cncn1 N1(C(C2CN(C(C(CCC)CCC)=O)CC23CCC3)=O)CCCC2(CCCC2)C1 C(C(CCC)CCC)NC(C1C(NC(CCOCC#C)=O)CC1)=O CN1CCC(CO)(CNC(=O)C(CC2CCC2)NC(c2cccc(=O)o2)=O)C1 CC(C)CCCC(C)CNC(=O)CC1C2CCC(C2)N1C(=O)C(C)C(C)(C)C c1(COC(C2CC3N(C)C(CC3)C2)=O)cc2ccc(F)cc2nc1Cl C(=O)(C(F)CCCC)NCC(CCCC)NC(=O)Cc1csc(S)n1 C(=O)(CCC(CC)CCC)NC(CC#CC)C(=O)NCC(O)C(=O)N(C)C c1(C(N2CCOC(COC)C2)CC(=O)NCCOCC)cncc2ccccc12 C#CCC(CC#C)C(=O)NCC(C)NC(c1cnccc1N(C)C)=O C(=O)(C(C)(C(C)C)OC)N(CC1CCN(C(C2C(C#C)C2)=O)CC1)CC c1(C(=O)NC(c2nnc(Br)n2C)C)ccccc1Cn1cccn1 C(=O)(C(CC(C)C)N(C)C(C1CCOCC1)=O)N1CCC(OCC)CC1 c1(C(C(=O)NCCCC2CC2)N(C(CSC)C)C)ccc(N(C)C)cc1Br c1(C(=O)NCC(N(C)C(c2cnc(C(C)(C)C)s2)=O)C2CC2)cccn(O)c1=O C(=O)(CC1=CCOCC1)N1C(C(=O)NCCC(O)CO)CC(O)C1 C1(CN(C(C2CC(=C)C2)=O)C)CN(C(c2ccc(-c3cnco3)cc2)=O)CCO1 CN=c1ccc(C(=O)NCCC2CCCN2C(=O)CNS(C)(=O)=O)c[nH]1 CN1CCC(C(=O)NCC2CCOC2(C)C)(NC(=O)CC2CCCC(=O)N2)C1 C1(NCc2ccc(OCCN(C)C)cc2)CC2CCC(C1)N2C C(=O)(CCCCCC#N)NCCC(C(=O)NC1C(CCOC)CCC1)OC C1(CNC(c2cc(C)c(Cl)s2)=O)CCC(C)CN1C(c1cn2ccnc2s1)=O c1(C(N(CC(C)NC(CCCC(=O)OCC)=O)C)=O)ccc2c(c1)COCC2 C1(C(=O)NCCC2(C(=O)NCCCC3CCCO3)CCC2)C2C3CCC(C3)C12 C(CC(C)(C)CC(=O)NCCC(O)CNC(c1cnn(C2CCC2)c1C)=O)OC c1(CC)sc(=N)[nH]c1C(N1CCC(C(C)NC(=O)C(C(C)C)N(C)C)C1)=O c1(CCC(=O)NCC(Cc2ccccc2)OCC)ccc(F)c2ccncc12 N1(C(C2(C#N)CC3CC3C2)=O)CCOC2(CCN(C(C3CC(=O)N(O)C3)=O)C2)C1 n1(CC)nccc1C=CC(N1CC(NC(c2cc(C)c[nH]2)=O)CC1CO)=O C=Cc1cc(C(=O)NCC(C)CNC(c2cccc(F)c2C)=O)cc(F)c1 N1(C(CC(C)N(C)C)=O)CCC(O)(C2CCN(C(C3CC3CF)=O)CC2)CC1 CCCCC(C)N=c1cc(C)nc(N(C(CC)CC)C)[nH]1 C1(COC)(NC(=O)CCCn2cccn2)CCN(C(=O)CC2C(=O)NN=C2C)C1 C1(NC(c2cncc(SC)c2)=O)CC(O)CN(C(=O)C(=Cc2cn(C)cn2)F)C1 CCC(C)(C)CC(=O)N1C[SH](CC2(O)CC(C(=O)NOCC(O)C(C)C)C2)C1 c1(CCC(=O)NC23CC(CNC(C(CC)NC(N)=O)=O)(C2)C3)ccc(Cl)c(C)c1 c1(C(=O)NCCNC(COc2cc(C)c(Cl)cc2)=O)ccc2c(c1)C(=O)NCC2 c1(CN2CC(C)N(C(C3CCCS3)=O)CC2)ccc(O)c([N+](=O)[O-])c1 Cc1cc(C)c(C(=O)NC2(CNC(=O)CC(C)C3CC3)CCCCC2)cc1N c1(CC)ncc(C(=O)N(CC(CC)NC(C2CC3CC3C2)=O)C)c(O)n1 NS(=O)(=O)CCCC(=O)NC1COCCN(C(C2CC2(F)Cl)=O)C1 c1(OC)cc(C(=O)Nc2ccc(C)c(C)c2)cc(Br)c1OC c1(CC(=O)N(C)CCNC(=O)C(F)=CCCF)c(F)cc([N+](=O)[O-])cc1F C#Cc1ccc(C(N2CCN(C(=O)C(C)c3ccco3)C(C)C2)=O)nc1 N1(C(CC=C(C)C)=O)CCC2OCCN(C(c3cccc4[nH]c(=N)oc34)=O)C2C1 CC1CCN(C(C2OC(C)CC2C)=O)C(C)C1NC(c1cc[nH]c1)=O C=CCCCC(N)C(=O)N1CCCC(O)(CC#N)CC1 N1(C(c2ccc(Cl)s2)=O)CCN(C(C2CCCCC(F)(F)C2)=O)C2(CCC2)C1 C1(C)(C(=O)NCC(N2CCCCCC2)C)CCCN(C(=O)CSc2ccsc2)C1 C1(CN(C(C2CCC(COC)C2)=O)C)CCCCN1C(=O)Cn1nc(C)cc1N C1(CCC)CCC(O)(C(=O)N(CC(C)NC(=O)C(O)C(F)(F)F)C)CC1 C#CCC(C)C(=O)NC1CC1CNC(=O)COCc1ccnn1C1CCOCC1 c1(CC(=O)NC(CNC(C(CC)(C)CO)=O)(C)C)cc(=O)oc2cc(C)ccc12 C(CCC(C)NC(=O)Cc1nocc1C)NC(C(c1cccnc1)OC)=O c1(C(N2CCCC(CNC(c3cc(=O)cco3)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 c1(C(C(=O)N(CCCNC(C2COC(=O)N2)=O)CC)(F)F)ncccc1F N1(C(C2C(CC)OCC2)=O)CCC2CN(C(c3cnccn3)=O)CC12 C1(CCC)CCCN(C(=O)N(c2c(I)ncn2C)CCN2CCOCC2)CC1 CC(O)(CNC(=O)C(F)OC(F)(F)F)NC(=O)COOC(F)(F)F c1(OCC)cc(C2(NCc3cccn3CSc3ccccc3)COC2)ccn1 c1(NC(CC)CNC(C2(C)CCOCC2)=O)ncnc2sc3ccccc3c12 c1(C(=O)NC(C)CN(C)C(C2(n3cnnn3)CCOCC2)=O)cnc(O)cc1O C(=O)(C(O)CNC(C1CC(C)(F)C1)=O)N(C)Cc1cncs1 c1(C(N(C)CC2N(C(c3ccn(CC)n3)=O)CCC2)=O)ccc2c(c1)OCO2 C1(COC(c2ccc(C(F)F)o2)=O)CCC(C(F)(F)F)C1 CCC(CCOC)C(=O)N1CC2CC2C1C(N1CCC(C(CC)CC)C1)=O c1(C(C(=O)NC(C)C)N(CC#N)CCN(C)C)nccc(Cl)c1Cl C12(C(N3C(C)(CNC(c4n(C)ncc4Cl)=O)CCC3)=O)CC1COC2(C)C C(=O)(C(C)CC(C)(F)F)NC1CCN(C(C2C(CC)CCO2)=O)C12CC2 c1(CN(CC=C)C)ccc(CNC(C2(NC(=O)CN3CCC3C)CCOC2)=O)cc1 Cc1ccnc(C)c1C(=O)NCC(C)CNC(=O)CCn1ncn(C)c1=O C(=O)(C(C(C)(C)C)C1CCC1)N(C(C)CNC(c1ncccc1Br)=O)C c1(CNC(C2C3CCCC23)=O)ccc2c(c1)CN(C(c1ccnnc1)=O)C2 c1(OC)nc(C(N2CC3(NC(=O)CCC4CC4(F)F)CCC2C3)=O)cc(O)n1 C1(NC(Cc2c(C)n[nH]c2C)=O)CC(C)CN(C(c2ccc(CO)nc2)=O)C1 CC(CCCCNC(=O)C(C)(C)F)NC(=O)CCC(=O)c1ccccc1OC(F)F CC1CC(C(=O)NCCN(C2CCCCC2)C(c2coc(Br)c2)=O)CO1 C(O)(C(F)(F)F)C1(CNC(C(N)c2cnc[nH]2)=O)CCC1 CCC(C)(C)CN=c1[nH]c(N2CCCC(CC(N)=O)C2)nc2cccc(F)c12 C1(CNC(CSc2c(C)n[nH]c2C)=O)CC(F)(F)CN1C(c1ncn(C)c1C)=O N1(C(c2n(CC)ccc2)=O)CCC(C)(C)C(C(=O)NCC(C)CC(C)C)C1 C12CCCN1C1CN(C1)C2=O.c1(CC(=O)NCC2COCCO2)cccnc1 Cc1cnn(C)c1C(=O)NC(C)(CNC(=O)CC1CC1(Cl)Cl)C(C)C N1(C(C(C)CC(=O)NC2C3CCCC23)=O)CCCC(NC(=O)CC2(C)CC2)C1 C(C(C)(C(=O)NCC1(F)CC(CNC(c2cc(N)ccn2)=O)C1)OC)OC Cc1nn(C)cc1C1=NOC(C(N2CCCC2CCNC(=O)C=C(Cl)Cl)=O)C1 c1(C(C)OCC)noc(C(=O)NCCN(C)C(C)=O)n1 C1(CC)CN(C(C2COC3(CCC3)C2)=O)CCN1C(=O)CSC(C)(C)C C=CCC(C)(C)CC(=O)N(CC(C)O)CCN(C(=O)CCCN1CCCC1)C(C)C CC(CC(C)(C)C)C(=O)NCCC1CCN(C(=O)C(F)(F)CN(C)C)C1 c1(C(N2CC(CNC(CCCOCC=C)=O)C(O)C2)=O)coc2ccc(F)cc12 C1(NC(C2CC3CCC2CC3)=O)CC2CC1CN(C(c1c[nH]nc1C(F)F)=O)C2 c1(CC)nc(NC2CC(CNC(=O)CCc3cnc(C)s3)C2)c(C)c(Cl)n1 N1(C(C(C)OCCC=C)=O)CCC(N(C(c2cc(CCCO)on2)=O)CC)C1 CC1CN(C(=O)CC(F)F)CC1NC(c1cc(N2CCCCC2)ccn1)=O c1(C(N2CCC(N3CC(C)(C4CCC4)C3=O)CC2)=O)cc2ccc(F)cc2s1 C(=O)(C#CC(C)(C)C)NC(C)C(CO)NC(C1COCCO1)=O c1(CCNC(C(C)OC(c2cc(C(F)(F)F)n[nH]2)=O)=O)ccccc1 Cc1ccc(OCCC(N2CCC(CN(C)C(C34CC(F)C3C4)=O)C2)=O)cc1C C1(NC(C(C)C2CC2)=O)C2CC1N(C(=O)Cn1cc(CO)nn1)C2 C(N=c1cc(NCC(CC)OC)nc[nH]1)c1ccc(-c2cccc(CC)c2)s1 c1(C(N2C(CNC(c3nnn(C)c3C(F)F)=O)CC2)=O)cc2cnn(C)c2s1 C1(=O)C(N(C)Cc2sccc2Cl)CCc2ccccc2N1.C(C(C)OC)SC.OC c1(CC2CN(C(=O)NCc3ncc(CC)s3)C2)cccc(C(F)(F)F)c1 N1(C(C(c2ccnn2C)C)=O)CCOCC(CNC(c2cncc(F)c2Cl)=O)C1 Cc1cc(CNC(C2CCC(CNC(=O)C(C)N(C)C)CC2)=O)ncn1 c1(CC(N2CCC(N(CCC)C(c3nocc3C)=O)C2)=O)ccc(C)c(C)c1 C1(C)(C(=O)NCC2(S(C)=O)CC2)CN(C(c2coc3c2COC3)=O)C(C)(C)C1 Cc1cc(NCC2CN(C(c3[nH]cnc3C)=O)CC2O)nc(C)n1 Cc1nn(CC(=O)NC2CC3CN(C(=O)Cc4cc[nH]n4)CC23)c(=O)n1C C(C(N=[N+]=[N-])C(=O)N(CCC(N1CCC(F)(C#N)C1)=O)CC)OCC N1(C(C=CCC)=O)CCC2(CCCCN(C(=O)Cc3csc(C)n3)C2)C1 C(=O)(N=c1c(Cl)c[nH]cc1I)C1CC(NCc2cc(OCC)cc(Br)c2)C1 c1(-c2cnc(C(NC)=O)nc2)ccccc1C#N.CC(C)CN(C)CCO c1(C(=O)NC(C(C)NC(=O)CCc2cccc(O)n2)CO)cccc2c1CCO2 C12(CNC(C3(C(c4ccc(Cl)cc4)O)CCNCC3)=O)CNCC1COC2 N1(C(C(C)=O)=O)CCC2(CCC2NC(C2CCNC(=O)C2)=O)CC1 c1(OCC)cc(Br)ccc1NC(=O)C(N1CC(O)C(O)C1CF)=O Cc1ccc(C(=O)NCC2CCC(NC(c3[nH]nnc3C3CC3)=O)C2)s1 c1(NC(C(C)Cc2cccc(F)c2)=O)cccc(S(=O)(=O)N2CCN(C)CC2)c1 C12(CNC(C(C3CCCCC3)N(C)C)=O)CC1CN(C(C1CCCOC1)=O)C2 CCCCCC(O)CC(=O)N(CCN(C(=O)CC(CC)C(F)F)C)C(C)C c1(C(C)=O)ccc(F)c(F)c1C.c12nc(cc(Cl)n1)C(=O)NC1(CC)CN2C1 CC(C)C(CN(C)C)C(=O)NC1CCN(C(=O)C(C)(C)F)CC1O C1(C(=O)NCCC2(C(N(CC(O)CO)CC)=O)CC2)CCCCS1 Cc1cc(F)cc(Cl)c1NC(=O)C(C1CCN(Cc2cccc(Cl)n2)CC1)C N1(C(=O)CCn2nc(-c3cccs3)oc2=O)S(=O)(=O)c2ccccc2S1 C1(N(C(c2c(C)snn2)=O)C)CN(C(c2cc(F)ccc2Cl)=O)CC1(C)C N1(C(C(=O)N(C)CC2CCCSC2)=O)CCOc2ccc(Cl)cc2C1 Cc1nnc2c(C(=O)NCC3(F)CC(CNC(=O)Cc4cn[nH]c4)C3)cccn12 Cc1ccc(CN(C=O)C(c2ccc(O)c(Cl)c2)C)cc1CO N1(CCC(=O)N(CCNC(=O)C(C)n2ccnc2)CC)CCP(C)(=O)CC1 C#Cc1ccc(C(=O)NC2(C)CC(NC(=O)CCC34CCC(CC3)C4)C2)o1 N1(C(C(C)OCC)=O)CC2(C1)OC1(C)CC2(NC(C2COCCN2C)=O)C1 S(=O)(=O)(c1ccc(=NCC2CCCOC2)[nH]c1)NC(c1cc(C)cc(C)c1)CC c1(C(N(C(C)C(=O)NCC2(CC(C)C)CC2)CCC)=O)cc(CO)oc1C N1(C(C#CCNC(Cc2c(C)non2)=O)=O)C2CCC1CC(C)C2 C(=O)(C(CNC(=O)C1=CCC(C)CC1)(CC)CC)N(CC#C)C c1(C(=O)NCC2(OC)CN(C(C3CN4CCN3CC4C)=O)C2)c(F)cc(F)cc1Cl c1(C(C)N(C(=O)C(F)(F)CC2CC2)C2CC2)ccc(CNC(=O)C(N)=O)cc1 Cc1c(Br)cc(Cl)c(NC(=O)CC2CCCN2C(c2ncccn2)=O)c1Cl C1(C(=O)NCCCNC(C2(c3ccn(C)c3)CC2)=O)CCC(C(F)(F)F)CC1 C1(C(=O)NC2COCCC2NC(C23CCC(CC2)C3)=O)CC2CCCC(C1)C2 C12CCCCN1CCN1CCC2C1.c1(N(S(C)(=O)=O)CC#N)scnc1C.CO N1(C(c2c(CC)ocn2)=O)CCCN(C(=O)CCN(CC(F)(F)F)CC)CCC1 c1(NC)cnccc1C(=O)NCC(F)CNC(C1OCCOC1C)=O N1(C(C2CCN(C)C2)=O)CCCCCC(NC(C2(CO)CCOCC2)=O)C1 Cc1cc(C(N2CC(O)CC2(C)C(=O)NC2CCC3(C(C)C)CC23)=O)nc(O)n1 N1(CC(=O)NC2(C)CC(NC(CC(C)O)=O)C2)C(=O)NC2(CCCCCC2)C1=O c1(CC)csc(C(=O)NC2CC(CNC(=O)CC(C)NC(=O)OC(C)(C)C)C2)c1 N1(Cc2scc(C(=O)Nc3c(OC)n(C)nc3C)n2)CCC(N=[N+]=[N-])CC1 CCS(=O)(=O)CC(=O)N1CCCC1(C(=O)NC1CC2(CC2)C1)C(C)C C1(C(=O)NC2CC(N(C)C(C3CC3(C)C(N)=O)=O)C2)CC2(C1)CC(F)C2 N1(C(C(C)(Cl)CCl)=O)CC2(CC(C(=O)NCC3CC3(F)F)CO2)C1 N(C(=NCCF)NC1CCN(C2CC2)CC1)Cc1cccc(C(C)O)c1 Cc1cc(C(=O)NCCn2cnc(C(=O)NCC(F)Cl)c2)nc(O)c1 C1(NC(Cn2nnc(C(C)(C)C)n2)=O)CC2(C1)CC2NC(C1CCC(=O)NC1)=O N1(C(c2c(OC)nn(C)c2)=O)CC2CCCC2(NC(c2cocn2)=O)C1 Cc1cc(C(N2CCCN(C(=O)C(C)NC(N)=O)CC2C(C)C)=O)c(O)nc1C CC1(C)CN(C(=O)C2CC2)CCN1Cc1c[nH]c2ccccc12 N1(C(C(C)OCCOC)=O)CCC(NC(C23CCC(CO)(CC2)C3)=O)C(CO)C1 c1(CNC(C2ON=C(C)C2)=O)ccc2c(c1)OCO2.C12CCN(C1)CCNC2=O c1(OC)cc(N(CCCNC(C2CCCC(C)C2)=O)C)c(F)cc1[N+](=O)[O-] C1(C(=O)NCC(CN(C)C(c2csc(C3OCCO3)c2)=O)O)CCCCS1(=O)=O CC1CCCN(C(c2cc(C3CCOCC3)nn2C)C(=O)NC2CC2)CC1 N1(C(C2(COC)CCCCC2)=O)CCC2C(CCCN2c2ncc(I)cn2)C1 C1(CC(=O)NCC2(O)CN(C(c3cc(CCC)on3)=O)C2)(CC=C)CCCCC1 c1(CC)cccc(C(=O)NCCNC(=O)C(C)(CC)OCc2ccccc2F)c1N C(=O)(C1=Cc2ccccc2OC1)N1CC(NC(c2cc(Br)cs2)=O)C2C1C2 C1(NC(c2cc(C)oc2C)=O)CCN(C(C2CC(=O)NC2(C)C)=O)CC1CO c1(CC(N2CC(CNC(C=Cc3nnn(C)n3)=O)C2)=O)cc(C(F)(F)F)cc(Cl)n1 c1(OC)cc(F)c(C(N2CC(NC(c3cncc(F)n3)=O)C2)=O)cc1OC N1(C(C(C)=C(CC)C)=O)CCOC(C(=O)NCC(C)(C)C(C)O)C1 N1(C(CNC=O)=O)CC2CC2(CNC(C2CCC2c2nc[nH]n2)=O)C1 C1(C2CC2)(CNC(=O)CC2CC2C(F)(F)F)CCN(C(c2ccon2)=O)C1 c1(C(=O)NCCCN(C(C(C=CC)O)=O)C2CC2)nccn2nccc12 N1(C(CN(S(CC)(=O)=O)C)=O)CC(F)(F)CC1CNC(c1nocc1C(C)C)=O c1(CCNC(c2ncn(C)c2)=O)c[nH]c(=NCc2c(Br)ccnc2Br)s1 C(=O)(CCC(=O)CC(F)(F)F)NC(=O)NCC1(C)CC1.CC1(N)C=CCS1 CCC(O)C(C)C(=O)NC1CC(F)(CNC(c2cnn3ccsc23)=O)C1 c1(C(=O)OCC)ccc(OCCNCC2NCc3ccccc32)c2cnccc12 c1(C(=O)NC(CNC(c2ccc(COC)s2)=O)C)cn2c(n1)CCC2 C1(NC(CCCC)=O)CCN(C(C2CCOC2C)=O)CC1 N(C1CN(C(=O)C=Cc2cccs2)Cc2ccccc21)C(C1(C)CC1)=O N=c1[nH][nH]c2cc(CN3CC4C(C(=O)NC(c5ccccc5)C#N)C4C3)ccc12 Cn1nccc1C(C(=O)O)N(C1COC1)C(c1ccccc1)=O c1(CNC(NC(C=C)C)=NCC2CC(S(C)(=O)=O)C2)cc(F)c(C#N)cc1C C1(NC(c2c(C)cco2)=O)C2CN(C(=O)CC3CCCC3C)CC12 C(=O)(C(O)CC(N)=O)NC1CC(NC(CCNC(COC(C)(C)C)=O)=O)C1 N1(C(c2ccc(C(OC)OC)o2)=O)CCC(NC(=O)C(O)CC(C)C)C(C)C1 Cc1nc(C)c(C(=O)NCC2(C(=O)NC3CCCC3C)CC2)s1 CC(C)CC(F)(F)C(=O)N(C(C)CN(C(=O)C(c1cccc(F)c1)N(C)C)C)C C1(CC(N2C(C)C(NC(=O)CCSCC(N)=O)CC2)=O)CC2(CCC2)CO1 C1(C(=O)NC(CC)Cn2cncn2)(CNC(=O)COCC(=O)OC)CCCCC1 N1(C(CNC(C2(SC)CC2)=O)=O)CCC(CC2CC2)CC1.C12CCC1C(=O)N2 c1(N(CC(CC)CC)C2CC2)ncnc(NC(C)CCc2ccccc2)c1C C1(NC(C(C)C2CC2)=O)CC2(C1)CC(NC(=O)C=CC1CCCCC1)C2 c1(C(N(CCN(C(C(COCC)C)=O)C)C)=O)cncc2ccncc12 N1(C(CSSC)=O)CC23CCCC2(C1)CN(C(=O)C(C(C)C)NC(N)=O)C3 c1(C(C(=O)NCC(CO)NC(C2N(CCC)CCC2)=O)(C)C)ccc(C#N)cc1 N1(C(CCN(C)CCO)=O)CCC(NC(=O)CC2CC(N(C)C)C2)CC1 c1(CN2C(CC(=O)NC3CNC(=O)N3)CCC2)nccc(OC2CCCCC2)n1 Cc1cccc(Br)c1NNC(=O)NCC1CCC(C)(C)CO1 C(=O)(C#CC1CCOC1)NC1CN(C(C(C)CSc2ccccc2)=O)CC(F)C1 C(=O)(C(C)CS(C)(=O)=O)NCCCC1CCN(C(C(n2c(C)ncc2)C)=O)CC1 C1(OC)C(NC(=O)C(C2CCCN(C(=O)CCc3ccncn3)C2)C)CC1(C)C C12(CC(N3CC(CCC)OCC3)=O)CCC1CN(C(C1(CC)CCCC1)=O)C2 N1(C(Cc2c(C)ncs2)=O)CCC(O)(C(C)NC(=O)C=Cc2ccccc2)C1 C(=O)(C(O)CC(F)F)NC(CCCC)CNC(=O)C=Cc1cc(C)no1 Cc1cccc(C(=O)N(C2CCN(Cc3cnc(O)c(Cl)c3)C2)C)c1Cl N1(C(COCc2n(C)ncc2)=O)CCC(C=CC(N2CCCC(C)(C)C2)=O)CC1 C1(CCNC(N2CCC(O)(C(F)F)C2)=O)CC2C=CC1C2 N1(c2cccc(C(C)=O)n2)CCS(=O)(=O)C(C)(C)C1 c1(CC(=O)NC2CC(NC(=O)CC34CCC(CC3)C4)C2)cc(O)nnc1O c1(OCC(=O)NC)ccc(-c2cscc2C(=O)Nc2ccc(C)cc2Br)cc1F C(=O)(CC(O)C(=O)NC1CC1NC(C1CCC1)=O)OC(C)(C)C c1(C(N2CCN(C(CCSCC)=O)C(CO)C2)=O)ccc2nc(O)oc2c1 c1(C(=O)NCC(C)(CO)NC(C2CCC(=O)N2)=O)cc(Cl)c(Br)[nH]1 CC(CC(=O)N(C)CC1(NC(=O)CN(C(=O)C(C)C)C)CC1)NC(N)=O C1(NC(CCN(C)C2CC2)=O)(CO)CCN(C(=O)C(CO)NC(N)=O)CC1 C(=O)(C(CC)C(C)C)NCC(C(=O)NCC(C#C)C(C)C)N(C)C C1(C)(NC(C2CN(C)C2)=O)CN(C(=O)C=CCN(C)C)C1 CC(C)CC(O)C(=O)N1CCOC(CNC(C2CN(C)CCO2)=O)C1 C(=O)(CS(=O)(=O)c1ccccc1)NC1C(C#N)CN(C(=O)CCc2cccs2)C1 c1(C2C(=O)N2)cncn1C.C1(CCN(C)CCO)CCCOC1.C1CCC1 c1(C(N2CC(C(N3CCN(Cc4n(C)cnn4)CC3)=O)C2)=O)cnc(Cl)c(Cl)c1 Cc1ccc(C(=O)NCC(C)(C)CCNC(=O)CC2CCC(C)C2)c(C)c1 c1(C(=O)NCC2CCC(NC(C3C(OCC)C3)=O)C2)cccc2oncc12 N1(c2ccc(CNC(C=C)C3CC3)cc2)C(=O)c2ccccc2C1=O c1(CNCC(c2ccccc2)O)ccc(OC(F)F)c(F)c1 C1(CC(=O)N(CC(C)CNC(=O)CC2(C)CC2)C)CC2CCC(C1)N2C CC1(CNC(C2(Cl)CC2)=O)CCCN(C(=O)Cn2ccccc2=O)C1 CCC(Cc1ccccc1C)C(=O)NC1(C)CC(NC(=O)CC(C)COC)C1 C1(C(=O)NC2CC(C)(NC(C34CC(F)(C3)C4)=O)C2)CC2(CCOCC2)CO1 c1(CC)cc(C(=O)C(N2CC(CC(=O)O)OC(CC)C2)C(=O)OC)ccc1C C1(CC)CN(C(=O)CC23CC(C2)C3)CCN1C(c1ncoc1-c1ccon1)=O N1(C(C2N(C(c3ccc(=NC)[nH]c3)=O)C3C(O)CC2C3)=O)CC(=O)N2CCCC2C1 c1(CN2C(CC#N)CN(C)C(=O)C2)ccc(C(=O)O)c2ccccc12 Cc1cccc(C(=O)NCC2CC(CNC(=O)CC3CC3)CO2)c1O c1(C(=O)NC2(CCOC)CCN(C(c3nc(Cl)c(Cl)s3)=O)C2)cc(C)nc(C)c1 C1(C(=O)Nc2ccc(O)nc2)CCCCN1C(=O)C(=O)Nc1cn(C2CC2)nn1 C1(CN(C)C(c2ccc(CO)nc2)=O)CCN(C(C2(C)CC2F)=O)CC1 N1(C(C(C(COC)C)C)=O)CC2CCCC(C1)N2C(C1(Cl)CCCCC1)=O c1(C(C)C)n[nH]cc1C(=O)NCC1CCCC1NC(=O)CC(=O)Nc1nccs1 c1(C(=O)NCC2CN(C(C(COC)OC)=O)CC2C)[nH]c2ccc(C)cc2c1Cl c1(CC)nc(-c2cccc(-c3ccc(C)nn3)c2)n(CCc2ccncc2)n1 CCC(CC)(CCNC(=O)C(c1ccccc1)=O)NC(=O)CCc1nccs1 c12cc(OC)c(cc1F)NC(=O)C1(C)CCN21.c1(C(=O)N)cc2ccccn2n1.CO C1(CNC(c2cc(O)n[nH]2)=O)CCCCN1Cc1ccc(F)cc1 C1(C(=O)O)CCCC(CNC(c2cc(-c3ccc(Cl)cc3)ns2)=O)CC1 Cc1cnc(C(=O)NCC2(NC(=O)CC(C)N(C)C)CCCC2)c(C)c1 C1(NC(CC(C)C)=O)CN(C(c2cccc3nc[nH]c23)=O)C2(CCOC2)C1 CCCCC(CC)CC(=O)N1CC(NC(c2cc(CC)nn2C)=O)CC12CCC2 N1(C(Cn2c(C)nnn2)=O)C(CNC(=O)C=CC2CCC2)CC2CCCCC12 Cc1c(NC(=O)CC2CCCN2c2cc(O)ncn2)cnn1C(F)F c1(C(N)=O)ncccc1NC(C1CC(F)CN1Cc1ccc(I)o1)=O C(CC(C)(C)NC(C1CNC(=O)O1)=O)=CC(=O)NCCN(C)CCF C1(NC(C(CCC(=O)OC)C)=O)CCC12CCN(C(C1COCC1(C)C)=O)CC2 C(=O)(C(C(F)(F)F)C(F)(F)F)NCCN(C(=O)Cc1c[nH]nc1O)CCO N1(C(c2[nH]cc(C)c2C)=O)CC2(CCN(C(C3CC34CCSCC4)=O)C2)C1 Cc1nn(C)c(F)c1C(=O)NCc1ccc(C(C)NC(=O)C(C)C(C)(C)C)cc1 C1(CNC(C(N2CCCCC2)C)=O)CN(C(=O)CCF)CC(C)(C)O1 Cc1cc(CNC(C2CC2C(=O)N(c2cc(C)ccn2)C)=O)nc(Cl)c1 c1(CCC(=O)OC)ccc(C(=O)NCCC(O)CNC(C2(O)CC(C)(C)C2)=O)cc1 N1(C(C(C(C)C)CO)=O)CCC2(CC1)CN(C(C1CCS(=O)(=O)N1)=O)CCO2 c1(CC(N2CC3C(NC(c4c(C)n[nH]c4)=O)(C3)C2)=O)ccc(Br)cc1F C(=O)(CCCCC(=O)NC12CC(NC(=O)CCCSC(C)(C)C)(C1)C2)NC c1(CC2N(C(=O)NC3C(C)(C)CCCC3)CCC2)ccc2c(c1)OCCO2 C#Cc1ccc(C(C(=O)NCCC=C)N(C)CCOCc2ccccc2)c(F)c1 CCCCCC=C(C)C(=O)NCc1ocnc1CC1CC2CC2C1 CC1(C)CCCC(CNCc2c(C3CN(C(C4C5CCCCC45)=O)C3)ocn2)C1 c1(OC)ccc(CC(N2CCN(C(c3occc3Cl)=O)CC2C)=O)c(F)c1 Cc1ncc(C(N2CC3CC(NC(C4CN(C(C)C)C4)=O)C2C3)=O)cc1N n1(CCSC)nnnc1C(C1(C)CCCO1)(C)NCc1ccnn1CC1CCC1 Cc1cc(CC(=O)NCC(CO)NC(C2CC3(CCC3)C2)=O)cc(F)c1 C1(C(N2CC(N(C(c3ccc(NCCOC)cc3)=O)C)C2)=O)CCCC(C)(C)C1 C(CC(C)(C)CC(=O)N1CC(NC(c2ccn(C3CCCC3)n2)=O)C(C)C1)OC N1(C(C(C(C)C)CO)=O)CCC(F)(F)C(CNC(c2cnc[nH]2)=O)C1 C1(CC(=O)NC(CN(C(CSCC)=O)C)(CO)CO)CSc2ccccc2O1 C(CCCCC(=O)N1CCC(CCNC(C2CC(C)CCO2)=O)C1)OC C1(C(=O)NCC(C2CC2)OC)CCCN1C(C)=O.c1(C2C(C(=O)NC)C2)ccccc1 Cn1nnc2c1C(C(=O)NCC1(NC(=O)C3CC3)CCOC1)CCC2 C=CCCC(C(=O)N1CC(C(=O)NCC)C1)NC(C1CCN1C)=O N1(C(=O)Cn2cc(C3CCCOC3)nn2)CCC(Cl)=C(Cl)C1 N1(C(CN2C(C)CCC2)=O)CCOC(C(N2CC(C(C)(C)C)C2)=O)CC1 C(=O)(C(C)(C)CO)NC(C)C(CO)NC(=O)Cc1cccc(C(F)(F)F)n1 N(C1COCc2ccccc21)C(N(C)CCOc1ccccc1)=O.C1CC1 N1(C(CN(C)C)=O)CCC2(CCC2NC(c2cncc(C(C)(C)C)c2)=O)CC1 c1(C(N2CC3C(CNC(c4c(C)ccnc4)=O)(C3)C2)=O)cc(C(F)F)ccc1Cl c1(OC)cc(F)c2c(C(=O)NC(C)(CNC(C3(F)CC3C)=O)C(C)C)n[nH]c2c1 N1(C(C2(C)CCN2C(=O)Cc2cc(Cl)c(Cl)[nH]2)=O)CCC(C(F)F)CC1 CN1N=C(CC(=O)N2CC(C)(NC(c3cn(C)nc3-c3ccco3)=O)C2)CC1=O N1(CC(=O)NC(C)CN(C)C(C2CC3CC2C3)=O)CC2C=CC1C2 c1(OC)cccc(C(N2CCCCC2CN(C(=O)C(C)C(C)O)C)=O)n1 c1(CC)cc(C(=O)NC23CC(NC(=O)C(CO)C(C)C)(C2)C3)ccc1OC c1(C(=O)NCC2CC(C)CN(C(C3CC3(Cl)Cl)=O)C2)ccc2n[nH]cc2n1 C1(c2onc(C(COC)CN)n2)CC12CCOc1ccc(Cl)cc12 C(=O)(C(O)C(CCC)NC(=O)C(C)OCC)N1CC(C#C)N(C)CC1 c1(C(=O)NC2CCN(C(C=C(CCC)C)=O)CC2C)coc2cccc(Br)c12 C1(NC(C2C(OCC)CC2)=O)CC(C)(CNC(c2cncs2)=O)C1 N1(CC(=O)N(C(=O)CCc2ccsc2)C2CC2)CCCC(c2ccccc2)CC1 c1(C(N(CCOC)CCNC(c2[nH]ccc2C2CC2)=O)=O)cccn2cnnc12 c1(C(=O)NCCCCC2CN(C(c3csc(Cl)n3)=O)C2)cnc(O)c(F)c1 C1(NC(C(C)(O)C2CCC2)=O)CCN(C(c2cn(CC3CC3)nn2)=O)CC1 c1(C(=O)NC(C(C)NC(c2cc(C)oc2)=O)C)ccn(C(C)C)c1C C1(CNC(C2CCCCC2)=O)CCCC1NC(C1CC=CCC1)=O CCN=c1[nH]c(C(=O)N(C2CCN(C(c3csc(Cl)n3)=O)CC2C)C)cs1 N1(C(C(C)(C)N(C)C)=O)CCC(C)(C(=O)NC2CCOC2(C)C)C1 C1(NC(c2c(C(N)=O)csc2)=O)CCN(C(c2coc(C3CCC3)n2)=O)CC1F C1(CC(=O)OC)Cc2ccccc2CN1C(=O)Nc1ccc2ccn(C)c2c1 C#Cc1cccc(C(=O)NC(CO)C(C)NC(C2(CC(F)F)CCC2)=O)c1F C(=O)(CCCC(=O)NCC(C)CNC(c1oc(CC)nc1C)=O)NCC c1(C(=O)NCCN(C2CCCC2)C(C2OCC(C)C2)=O)cnn2c1CCCC2C N1(C(CC=C)=O)CCC(NC(=O)CC2CCOC2(C)C)CC(O)C1 C1(CNC(c2ccnc(S)c2)=O)CCN(C(=O)C(O)C2CCCC2)CC1O Cc1ccccc1NC(c1cccc(CSC)n1)c1nnnn1C1CCCCC1 N1(C(C2C(CC)C2)=O)CC(NC(c2cncc(C)n2)=O)CC2(CCC2)C1 c1(C(=O)NCC(C)(C(C)C)NC(c2nc(C)oc2)=O)cccc(F)c1C#N C(=O)(C(C(C)(C)C)N1C(=O)CCC1=O)N1CC(NC(C(COC)(C)OC)=O)C1 Cn1cc(C(N2CC3C(C(=O)NCc4ncc[nH]c4=O)C3C2)=O)ccc1=O C1(NC(c2n(C)nc(CNC(=O)C(F)CC3CCC3)c2)=O)CCCC2(CC1)CC2 C1(C(=O)NC(CC(=O)N(C2CCN(CC)CC2)C)(C)C)CC(=O)OC1(C)C C(c1c(C)noc1C)=CC(=O)NC1CC(CNC(C2(COC)C=CCC2)=O)C1 CC1(C)C(NC(=O)C=Cc2cc[nH]n2)CCN1C(=O)CCC(=O)NC1CCCC1 C1(NC(C23CC2C3)=O)CCN(C(=O)C2=CCCCC2)CC1F N1(C(CC2CCN(C(C3(C)CCCC3O)=O)C2)=O)CCCC(F)CC1 C(CC(C(=O)NC(C)CC(=O)OC)NC(=O)C(C)=CC(C)(C)C)SCC c1(N(C)C)ccc(CNC(C2C3CC3CN2C(C2CC2(Cl)Cl)=O)=O)cn1 N1(C(c2cc(C)nn2C(F)F)=O)CC2CC1CN2C(=O)COC(F)(F)C(F)(F)F C1(NC(=O)CCF)CN(C(c2ncccc2Br)=O)C2(CCCOC2)C1 Cc1cccc(C)c1C(=O)NCC1CC1C(=O)NCC1CN(C)CCN1C c1(-c2c(CNC(C3COC4(CNC4)C3)=O)c[nH]n2)cccc2ccccc12 C(=O)(C(F)(F)C(F)F)NC1(CN(C)C(c2cc(-c3ccccc3)co2)=O)CC1 N1(C(COC(CC)(C)C)=O)CC2CC1CN(C(=O)C(=O)Cc1cccc(F)c1)C2 c1(C(N2CCC(O)C2c2cccc(F)c2)=O)c[nH]cc(F)c1=O CC1(F)CCN(C(C2CC(O)CN2C(c2cccc(Cl)c2)=O)=O)C1 c1(CC)cc(C)c(C(=O)NCCN(S(=O)(=O)CC)C)o1.C12CN(C1)C(=O)CS2 CC(C)C(O)CC(=O)NCc1occc1C(=O)N(CC(=O)NC1CC1)C C(C(CC(F)(F)F)NC(c1csc2nccn12)=O)NC(c1csc(CO)n1)=O CC1CC(NC(c2nc(Cl)ccc2Cl)=O)CCN1c1ncc(C(C)(C)O)cn1 C1(C(N2CC(OC)C(NC(=O)Cc3cc(C)nn3C)C2)=O)Cc2nc(C)cn2C1 N1(C(C(C)C)=O)CCC2(CNC(=O)C(c3ccc(F)c(F)c3)(C)C)CCCCC12 CCCS(=O)(=O)CC(=O)NC1CN(C(c2cnccc2Cl)=O)CC1C C1(CCC(=O)NCC(F)F)CCN(C(=O)C(N2CCCC(F)C2)=O)CC1 c1(NC(N)=O)cccc(CC(=O)NC2CCC2NC(c2ccc(CO)cc2)=O)c1 O=C(CC(F)(F)C(F)(F)F)NCC1(C2CC2)CCN(C(=O)CCn2cncn2)C1 c1(CC)ccc(C(=O)NCC(O)CN(C(=O)Cn2nc(C)oc2=O)C)nc1 N1(C(C(C)Oc2cccc(C)c2)=O)C2CCC1CC(CNC(C1CC1C)=O)C2 CC(CCN=c1cc(Cl)nc[nH]1)NC(c1ccn2c(O)nnc2c1)=O C1(C)(C(=O)NC(C=C)C2CCC2)CCCN1C(C1CCCSC1C)=O Cc1nc(CNC(=O)C(n2cc(CC3CC(F)(F)C3)nn2)C)nc2ccccc12 C(=O)(CCCS(C)(=O)=O)NC(C1CCN(C(C2(C(F)F)CCC2)=O)C1)C Cc1cccc2c1CCOC2C(=O)NC1(CF)CCN(C(=O)CSC)C1 c1(NCCC2N(C)CCC2)nccc(=NCc2ccnc(C#N)c2)[nH]1 C1(CC(=O)NC(c2nc(C)[nH]n2)(C)C)C2CCCC2N1C(c1ccc(C)nc1)=O N1(C(C2ON=C(C)C2)=O)CCC(O)(CN(C(=O)CCc2c(C)noc2F)C)C1 N1(C(C(COC)OC)=O)CCC(=CCNC(c2coc(C3CCC3)n2)=O)CC1 c1(N2CCCC(CNC)C2)nc(=N)[nH]c(=NCCc2c[nH]nc2O)[nH]1 C1(c2onc(C(C)C)n2)CCCN(C(=O)C(=O)N(CC)CC2(O)CCNCC2)C1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(C2CCCCO2)=O)C(C)(C)C1 c1(OC)ccc(C2(C(=O)NCCCCCCN(C(=O)C(C)OC)C)CCC2)cc1 Cc1ccc(F)c(C(N2C3CCC(C3)C2C(=O)N(CCCO)C2CC2)=O)c1F C1(CN(C(C2CCC(NC(C(CO)NC(=O)OC)=O)C2)=O)C)CCC(C)CC1 c1(OC)cc(NC(C2CCC(C)N2Cc2ccc(F)nc2C)=O)c(Br)cc1Br c1(C(N2CCC(C(C(=O)NC(c3cccc(O)c3)C)(C)C)C2)=O)ccc(C#N)n1C C1(CC(=O)NC(CN(C(C2(C(=O)OC)CC2)=O)C)C)CSCCS1 c1(NC(=O)NC2CC2C(=O)NCc2c(COC)cccc2)ccc2n[nH]cc2c1 c1(C(C2CC2)NC(N2CCC(c3ncc(C(=O)OC)s3)C2)=O)ccc(N)cc1C C1(C(=O)NCC(CCC)C)C=CCN(C(C2(OC(C)=O)CC2)=O)C1 c1(CCC(=O)NC2CN(C(C3C(OC)CCCC3)=O)C2)c(C)nc(SC)nc1O CC(C)C(CNC(=O)C=CCn1cncn1)NC(c1n[nH]cc1C(F)(F)F)=O C1(F)(CNC(Cc2nc(C)sc2C)=O)CCCN(C(=O)C=CC2CC2)C1 c1(N2CC(C)(NC(C(C)C(C)c3ccc(F)cc3)=O)C2)ccc(C)c(C)c1 c1(C(N2C3CN(C(Cc4c(C)noc4)=O)C(C3)C2)=O)ccc2nc[nH]c2c1 C(C)(C(C)NC(N1CC(N(C2CCC2=O)C(C)(C)C)C1)=O)(C1CC1)OC C1(C(N(CCCNC(c2c(N)nccn2)=O)CCO)=O)Cc2c(F)cccc2O1 c1(C(N2C(CC)C(OCC(=O)OC)CC2)=O)cnn2ccccc12 c1(C2CN(C(C(c3cn(CCOC)nc3)=O)=O)C2)cc(F)c(Cl)cc1C C1(COC(C)C(=O)NCCN(C(C2(C(F)(F)F)CCCO2)=O)C2CC2)CCCCO1 C1(CN(C(c2cn(CC)nn2)=O)C)CCCN(C(=O)CSCc2ncc[nH]2)C1 CC1CC(C(N2CCC(N(C(=O)CCc3ccnn3C)C)CC2)=O)CC(C)(C)C1 N#Cc1c[nH]c(NC2CC23CCN(C(=O)OCc2ccccc2F)CC3)nc1=N C1(NC(C=Cc2ncn(C)c2)=O)CC2CC1N(C(C1(C)CC1(Cl)Cl)=O)C2 c1(C(=O)NC2CN(C(=O)CCCCBr)CC(F)C2)n[nH]c2cccnc12 CCC(CC)C(=O)N(C1CCC(NC(=O)CC(c2cccs2)NC(N)=O)CC1)C c1(OC(C)C)cnc(C(=O)N(C2CCCC2)CCNC(=O)C(O)CN(C)C)cn1 C(C(C)(C)C(=O)NCC1(F)CCN(C(C2CC(=O)N(C)C2)=O)C1)OCC C1(C(=O)NC(C2CCOCC2)C)(CC)CCN(C(=O)C(C)SC(C)C)C1 C(=O)(CC(C)C(=O)N(CC(C)N(C(=O)Cc1ccc(C)nc1)C)C)OC c1(C(C(=O)NC)N(C2CC2)Cc2cccc(CO)c2F)cc2ccccc2o1 C1(CNC(c2c(C)nc(O)s2)=O)CC12CCN(C(C1CC(C)(F)C1)=O)CC2 CC1(C)CC(NC(c2nnnn2Cc2ccc(F)cc2)c2cn[nH]c2)C12CCC2 c1(CC)nc(N2CCC(C)(NC(=O)CCOc3ccc(F)cc3)C2)cc(C)n1 N1(C(Cc2c(C)cco2)=O)CC(C)CN(C(c2n[nH]c(=N)[nH]2)=O)C(C)C1 N1(C(CS(=O)(=O)NC)=O)CCC(CNC(c2ccc(S(C)=O)cc2)=O)C(F)(F)C1 N1(C(C(CC=CC)NC(=O)OCC)=O)CCOCC(CO)C1.C1(=O)CN1 c1(C(N2CCOCC(C)(C)C2)=O)ccc2c(c1)S(=O)(=O)NC=N2 C(C(COC)CC(=O)NC1COCC1C(N1CCC1C(N)=O)=O)OC N1(C(=O)NCC(C)S(N)(=O)=O)CC2(C)CCC2(C)C1 C1(CC(N2CC(NC(C3CCC(=O)NC3)=O)C2)=O)CC2(CCC2)CCO1 N1(C(CC)=O)CCC(C2CCCN(C(c3ccc(COC)nc3)=O)C2)C1 Cc1nc(C(C)C)cc(NC(c2ncccc2F)C2CCCCCC2)n1 c1(CNC(C(=O)NC(c2ccnn2C)CC)=O)cccc2c1OCCCO2 C(N=c1[nH]cnc2c1COC2)C1N(C(C2CCCC(C)C2)=O)CCC1 c1(OCC(N2CC3(C(=O)NC45CSCC4C5)CC2CO3)=O)ccc(F)cc1F C(=O)(CC(C1CC1)NC(C)=O)NCCN(C(C(c1cnn(C)c1)OC)=O)C N1(C(CCC=CC)=O)CCC(NC(=O)COC(C)CC)CC1C c1(SCC)ccccc1C(=O)N(C)CC1CCCN1C(=O)CCc1cnn(C)c1 CCCCCC(O)CC(=O)NC1CC2CN(C(C34CC3C4)=O)CC2C1 C1(C(=O)Nc2cccc(NC(C34CCCC3CCC4)=O)c2)CCc2c[nH]nc2C1 N1(C(C(C=C)OC)=O)CCC(C2CC2)C1C(=O)NC(COCC)C(C)C CC1(c2ccccc2)COCCN1C(c1ccc(F)c(C2CC2)n1)=O n1(CC)ccnc1C=CC(=O)NC(C1CCCC1)CNC(c1ncoc1C)=O c1(CNC(=O)C(C2CCC(F)(F)CC2)O)cn2c(n1)CCC2 C(CCC(F)(F)F)NC(C1CCCC(NC(c2ncccc2F)=O)C1)=O CC1(CNC(C2CCOC2CNC(=O)COCCF)=O)NC(=O)NC1=O CC1=NOC(=O)C1CCC(=O)NC1CC1CNC(c1cc(C)no1)=O N1(C(c2ccno2)=O)CCC(O)C(C(N2CCCC2c2cccnc2)=O)C1 N1(C(C(COCC)(C)C)=O)CCN(C(=O)CCC=CBr)C(CF)C1 Cn1cnnc1C1CCN(CC(NOCC(=O)N(C)C)=N)C1 c1(C(=O)NS(CCCC)(=O)=O)cc(Cl)ccc1C.C12C3CN(CC13)C2 c1(OC)ccc(S(=O)(=O)NC23CC(N)(C2)C3)cc1.c12ccc(cc1)C(OC)CC2 C=CCCCCC(=O)NC1CCN(C(c2nc(CC)oc2C)=O)CC1CO CCC(C)C(CC(=O)N(C)CC1CCCN(C)C1)NC(=O)C(C)(C)n1cccn1 C(C(C)CC(F)(F)F)NC(CN(C(c1c(CC)nco1)=O)C(C)C)=O c1(C(=O)NCCNC(c2ccc(Cl)c(OC(F)F)c2)=O)ccc(F)c(Cl)c1F N1(C(C(COCC)C)=O)CCCC2(CCN(C(=O)Cn3nc(CC)cc3C)C2)C1 c1(C(C)N(CCC(N2CC(O)(CO)C2)=O)C(=O)CO)ccccc1[N+](=O)[O-] c1(CSCC)ccccc1C(=O)NCC1CC1NC(=O)CNS(=O)(=O)NC N1(C(CNC(CCC(C)C)=O)=O)CCCCC(NC(C2CCCS(=O)(=O)C2)=O)C1 C1(NC(CNC(=O)NC)=O)CCN(C(C2CC2F)=O)CC1c1ccccc1 Cc1c(NCCCCC(C)C)ncnc1NCc1cccc(C(F)(F)F)n1 c1(OCC#C)cc(CN2CC3CC2C3C(=O)NCC(F)(F)F)ccc1OC c1(CC)nc(C)c(C(=O)NC2CC(NC(=O)C(c3cccc(Cl)c3)(C)C)C2)s1 C=CC1CN(C(C23CC2CCN3C(=O)CCc2cnn(C)c2)=O)CC1O C=CCC(C(=O)NCc1ccc(C(N2CCC(C3CC3)C2)=O)s1)C(C)C c1(CCC(N2CCOC(C3CCOCC3)C2)=O)ccc(O)nc1 N1(C(c2ccc(F)c(N)c2F)=O)CCC2(CCCN2C(=O)C=C2CCOCC2)C1 N1(C(CSCC#C)=O)CCC(F)C(NC(c2csc(-c3c[nH]nc3C)c2)=O)C1 n1(CC(=O)NC(C)CNC(c2ccc(N(C)CCO)nn2)=O)cc([N+](=O)[O-])cn1 n1(CC(=O)OCC)nc(C(=O)NC23C(CCN(C(C)=O)CC2)C3)c2c1CCOC2 c1(C(=O)NCC2(F)CN(C=O)C2)ccc(N)cc1Cl.C1(C2N(C)CC2)CC(=O)NC1 N1(C(C=CC(CC)=CCC)=O)CC(F)(F)CC1(C)CNC(=O)C(F)=C(C)C c1(OC)ccc2[nH]c(=NC3CCN(c4nncs4)C3)nc(N3CCC(F)C3)c2c1 N1(C(CCC(C)C)=O)CCCC2(CCCN2C(=O)CC2CCC(C)(C)CC2)C1 c1(C(=O)NCc2ccc(F)c(F)c2)csc(C2=COCCC2)n1 Cc1cccc2c1CN(C(C1(C3CC3)CN(C(=O)C(C)CC(C)(C)C)C1)=O)C2 c1(OC)ccc2nc(N3CCC(CCNC(C4CC4(F)F)=O)C3)c(C#N)cc2c1 N1(c2nccc(OCCC)n2)CC(NC(C2COCCO2)=O)CC12CCOCC2 c1(C(=O)NCC2N(C(C(C)OCC)=O)CCCC2C)cc2cccc(F)c2o1 C1(NCC23OCC(NC(N4CCC(N5CCC5)CC4)=O)(C2)C3)CCCC1C1CC1 c1(C(=O)NC(CNC(c2c(NCC)scn2)=O)C2CC2)ccc(C2CC2)nc1 N1(C(CC2C(C)(C)OCC2)=O)CCC(F)(C(=O)NCCN2CCCC2)CC1 c1(CCC(N2C(C)CN(c3nccc(Br)n3)CC2)=O)cc(F)c(F)cc1[N+](=O)[O-] C1(OC)CCCCC1C(N1CCC(N(C(=O)CCC2CC2C)CC2CC2)CC1)=O N1(CCC(=O)NCCN(C(C2C(CC)C2)=O)CC2CC2)CCNC(=O)C1 N1(C(C23N(C(C4CCSC4)=O)CC(C)(C2)C3)=O)CCCC2(C=CCO2)C1 c1(C(N(C)CC2CN(C(=O)CC3CC3(C)C)CCO2)=O)nccn2nccc12 C(=O)(C(C)S(C)(=O)=O)N1CC(OC)C(NC(c2nc(C)sc2Br)=O)C1 Cc1cccc(C)c1OCc1ncnc(N(CCCCC2CC2)C)n1.C1C(=O)N1 N1(CC)CC(NC(=O)CC(C)(C)N(C(=O)CC2OCCC2(C)C)C)C(C)C1 C(=O)(C(CNC(=O)C(=O)N(C)C)C(C)(C)C)N(C1CC1(C)C)CC c1(CC(=O)NCCCCCNC(C2(C)CC(=C)C2)=O)cccc(C(C)C)c1 CONC(=O)C(=O)NCC1CCCN(C(=O)CCN2CCCCC2)C1 C(CCCCC(=O)NC(C)(CNC(c1ncn2c1CCC2)=O)CO)OCC N1(C(Cc2cccc(OCC)n2)=O)CC(NC(=O)C(F)CC2CC2)CCC(O)C1 N1(C(C2C=C(C)CS2)=O)CCC(C(CO)NC(=O)C(C)Cc2cnc[nH]2)CC1 N#Cc1cc(NC(=O)CC2CN(C(c3cc(O)c(O)c(Cl)c3)=O)C2)ccc1Br C(=O)(C(C)(O)CC(F)(F)F)NCC12CCC(NC(CCC(=O)NC)=O)(CC1)CO2 c1(CN2CCCC(CNC(c3ccc(F)c(Br)c3)=O)C2)cc(F)c(O)cc1F C1(COC)(NC(=O)CCC(C)(C)C)CCCN(C(C2CC2c2ccccc2)=O)C1 C(=O)(CCC(C)(C)N(C)C)NCC(C)(CNC(=O)C(C)C(C)(C)C)OC C1(OC(C(=O)NC(C2CN(C(CN(C(C)=O)C)=O)C2)C)C)CCCCC1 C1(OC)CN(C)C(C)(C(=O)NCC2(NC(=O)C(C)=CC(C)C)CCCCCC2)C1 c1(C(C)(C)C)cccc(CC(N2CCC(C(=O)N(C)C)(CCO)C2)=O)c1 C1(C(N(C)CC2COCCN2C(C2(C)C=CCC2)=O)=O)CCCC(F)(F)C1 N1(C(COCC)=O)CCCC(C)(C)C1C(=O)Nc1ccc(N(C)C)nc1 C(=O)(CC1=CCN(C(=O)COCCF)CC1)NCCc1nc(CC)on1 C(CC(=O)Nc1cccc(F)c1C)(C(F)(F)F)NC(COCCCCC)=O N1(CC(N2CCC(C(C)NC(=O)C(c3cccnc3)C)C2)=O)CC(=O)N(C)C1=O CON1CCC(CC(=O)NC(CNC(c2cnnn2C2CC2)=O)C(C)C)CC1 CCCC(CN=c1[nH]c(N2CCC(Br)=C(C)C2)nc2c1SCC2)OCC C#Cc1nc(C(=O)N(C(CNC(C2CSCCS2)=O)C2CC2)C)cs1 C1(C)(NC(=O)NC(c2cccc(I)c2)C)CCN(Cc2ccccc2)C1 Cc1c(CC(=O)NCc2cc(C(=O)NCC3CCCC(O)C3)cs2)ncn1C N1(C(CCC(C)OC)=O)CC(NC(=O)C(C)(Cl)Cl)C2(CC2)C1 C1(CNC(C(C)=CC2CC2)=O)CCCCCN1C(C1CC2(CSC2)C1)=O N1(C(CCCCNC(C)=O)=O)CCC2(NC(C3CCC(C)C3)=O)CCCC12 N1(C(C(C)=CC2CC2)=O)CCCCC(N(C)C(c2ccc(F)s2)=O)C1 Cc1cc(C(N2CCC(NC(C3CC3(C)C)=O)C2C)=O)nc(O)n1 C1(C(=O)NCCCC2CCN(C(c3n(C)cnc3)=O)CC2)CCCCC(F)(F)C1 c1(C(=O)NC(C)CNC(c2cccc(=S)n2O)=O)cc2n(n1)CC(F)C2 N1(C(C2CC(S(C)(=O)=O)C2)=O)CCC2CCCC12CNC(c1ncccn1)=O C(=O)(CCCC(=O)N1CCC(NC(c2csc(C3CCCCC3)n2)=O)C1)OC N1(C(CCOC)=O)CC2C(C1C(=O)Nc1cc(Cl)c(C#N)cc1Cl)C2(C)C Cc1coc(C=CC(N2CC3CC3(NC(=O)CCCCN(C)C)C2)=O)n1 c1(C(N2CCCC(C)(NC(=O)CCP(C)(C)=O)C2)=O)cccc2ccsc12 CCCC(CNC(c1ccc[n+]([O-])c1)=O)C(=O)NCCc1nccn1C C1(NC(COCCC#C)=O)CC(O)CN(C(c2ccc(O)c(CC)c2)=O)C1 CC1CC(=O)NC(C(=O)NC2CC(NC(c3coc(C4CC4)n3)=O)C2)C1 C1(CNC(c2c(C)oc(Cl)n2)=O)CC(F)(F)CN1C(C1CN(CC(F)(F)F)C1)=O C#CCC(CC#C)C(=O)NC1CC2C(NC(=O)C(C)N3CC(C)C3)C2C1 CC(O)(CNC(c1cnc(C2CC2)s1)=O)CNC(=O)CCSc1nnnn1C c1(C(=O)NC2C3CN(C(C(C)OCC)=O)C(C3)CC2)csc2c(C)cccc12 C1(O)(CN(C(=O)CC2CCCSC2)C)CCN(C(=O)COC2CC2(F)F)CC1 c1(NC(CC(C)O)=O)nc2c(s1)CC(NC(c1ccnnc1O)=O)CC2 c1(C(=O)NC(C2CCOC2)CNC(C(=CC2CCCC2)C)=O)ccnc(C)c1C CCC(F)(F)C(C)(C)C(=O)NCC1C=CC(NC(c2ccc(=N)[nH]c2)=O)C1 CN1CC2(CC2)CC1C(=O)NC1CCC(C(=O)NCCCC2(C)CC2)CC1 N1(C(CCOC(C)=O)=O)CCC(O)(CN(C)C(C2(CF)CC(F)(F)C2)=O)C1 C(=O)(Nn1cnnc1C)C1(CF)CCN(C(C(C(C)(C)C)OC)=O)C1 N(C1CS(=O)(=O)Cc2ccccc21)C(c1noc2c1CC(C(=O)OC)CC2)=O C12(C(=O)NC3C(C)C3C)COCC1CN(C(=O)CC13CCCC1C3)C2 c1(C(=O)NC2CC(C(=O)Nc3cc(CC)c(C)cc3)C2)cccc2nccn12 N1(C(c2n(C(CC)CC)ncc2)=O)CC(NC(=O)C(C)(C)CO)CC12CCCC2 C1(CNC(c2c(C)cnnc2O)=O)CCCC2(CN(C(c3ccsc3)=O)C2)O1 c1(NC(=O)CC2CCN(C(c3cccc(O)c3F)=O)CC2)cnccc1[N+](=O)[O-] N1(C(C(c2scc(C)n2)C)=O)CCOC(C(C)NC(c2nccn2C)=O)C1 C1(C(N2C(C)CC(C#N)C2)=O)CC2CN(C(c3cc(C(F)F)[nH]n3)=O)CC2C1 CON(C(=O)C1CCCN(C(=O)Cn2ccnc2C)CC1)C1CCC1 N1(C(C(C)(C)c2cnc[nH]2)=O)CCOC(CCNC(=O)C=Cc2cc[nH]n2)C1 C(c1c(C)coc1C)=CC(N1CCC(C(CNC(C(CC)=CC)=O)C)CC1)=O C1(CS(=O)(=O)NC(C(CC)C)c2ccccc2)CCN(C(C2CC2(C)C)=O)CC1 C1(C(=O)NC2COC(C(F)F)C2)CCCCN1C(C1C2CCCCC12)=O c1(C(=O)NC(CC)CNC(C2CC=CC2)=O)csc(=NC2CCCCC2)[nH]1 C1(C(C)C)CN(C(C2CCC(CNC(c3ccc(O)nn3)=O)C2)=O)CCCO1 c1(C(=O)NCC(N2CCN(C(C(C)(C)CF)=O)CC2)=O)cc2c(cc1Cl)NCC2 CCCCCCC(C)C(=O)NCc1ccc(CNC(c2ncoc2CC)=O)cc1 N1(C(c2cncs2)=O)CCC(C2CC2)C1CNC(C1(O)CCOCC1)=O N1(C(CC(C(=O)OC)C)=O)CC2(C1)SCCC2NC(c1ccncc1F)=O C#CCC(C(=O)NC(CN(C)C)CC(C)C)NC(=O)CSc1ncccn1 CC(CC(=O)NCC1(F)CC(CNC(=O)C(C)S(C)(=O)=O)C1)C(C)(C)C C1(NC(C2(C)CCC(C)C2)=O)CN(CCOc2ccccc2)CCC1C N1(C(COC)=O)CCC2(C1)CN(C(=O)CN(C)S(=O)(=O)N(C)C)CCO2 c1(C(=O)NC2C(CC)CN(C(c3cnc[nH]3)=O)CC2)cccc2cncn12 N1(c2ncc(C)s2)CCCC(c2nc(CN(C)C)nn2Cc2ccccc2)C1 N1(C(c2c(OC)cccc2)=O)CCCCC(C(=O)Nc2ccc(O)c(F)c2)C1 N1(C(C2CCc3n(cc(C)n3)C2)=O)CCc2cc(Br)cc(F)c21 CCC(C)CCC(O)CC(=O)NCC1CCCCN(C(=O)C(C)(C)C(C)C)C1 c1(SCC(=O)NC2C=CCN(C(C3(C(F)F)CCCCC3)=O)C2)cccc(O)c1 C1(NC(c2c(C)cccn2)=O)CCCCN(C(=O)CSCc2cscn2)C1 c1(NC(C2N(C(c3ccc(C)nc3Cl)=O)CC(F)(F)C2)=O)ccc2ccoc2c1 c1(C(=O)NCC2C3CN(c4nccc(OC(F)F)n4)CC23)cncc2ccsc12 C1(CC)C(C(N2CC(C(C)OC)C2)=O)CCCN1C(c1scc(C)c1C)=O C(C(C)(C)C)=CC(=O)NCCCN(C(C1CC(C(=O)OC)C1)=O)CC O=C1NCCN(Cc2cc(F)cc(F)c2)C1c1ccccc1 C1(C2(O)CCOCC2)(C(=O)NC2C(NC(c3cc(C(C)C)on3)=O)COC2)CC1 C1CCCCC(=O)O1.CC(C(=O)OC(C)(C)C)SC(F)F Cc1cc(CN2CCCC(Cc3nc(C4CCCCC4)no3)C2)cc2c1CCC2 N1(C(c2c(C)oc(C)c2Br)=O)CCC2CCN(C(=O)CCCN(C)C)C2C1 c1(C(=O)NCCCCC(C)NC(CN(CCC)C)=O)ncn2c1CCCC2 N1(C(C2(C#N)CCCCC2)=O)CCCCCCC1C(=O)NCC1CC1 CC(C)CS(=O)(=O)CCC(=O)N1CCCC1C1CCCN1C(c1cccnn1)=O N1(C(C2(NC(C(C3CCCCC3)C)=O)CC2C)=O)CC2(CCOCC2)C1 N1(C(C2CCN(c3n(C)ccn3)C2)=O)CC2CC1CCC2NC(=O)CSC(F)F CC(CCC(C)(C)C)C(=O)N1CCCCC1CNC(=O)CCn1ccccc1=O c1(N2CCCC(NC(c3cc(C)ns3)=O)(CO)C2)ncc2c(n1)CCOC2 C1(NC(=O)NC2CCCCC2n2cc(CCCC3CC3)nn2)CC2(CCC2)C1 c1(C(C)(C)C)ccc(C(=O)NCC2CC2CNC(=O)C=C(Cl)Cl)cc1F C(CC(CC)C(=O)N1CC(O)(CCNC(=O)C(C(C)C)NS(N)(=O)=O)C1)=CC c1(CN(C(C2(C)C(C)C2)=O)C)cccc(CNC(C2CC23CCC3)=O)c1 Cn1ncc2c(C(=O)NC3C4CCC3N(C(C3CC35CCCC5)=O)C4)ccnc12 C1(CNC(C(C)CSC(F)(F)F)=O)CN(C(c2ccnn2C)=O)CCC1C c1(C(=O)NC(c2cncc(OC)c2)COC)cc2cccn2c(O)n1 CC1=CCC(C(=O)NC2CN(C(c3ccccc3-n3ccnc3)=O)CC2F)CC1 Cc1c(C(=O)NCC2CCN2C(=O)C(C)CC2CC2)cncc1Br C1(NC(C(C)NC(N)=O)=O)C=CC(C(=O)N(CC(F)(F)F)CC2(OC)CCC2)C1 CC1CCN(C(=O)CC2CC3(CC3)C2)C(C)C1NC(c1cnc(O)n(C)c1=O)=O C=CCN=C(NCCCCN1CCCC(CO)C1)NCC(c1ccccc1)(C)O Cc1cnc(C(=O)NC2CCC(CNC(=O)C(C)(C)c3ccnn3C)C2)nc1 C1(CN(C(N2CCOCC2C2CCCOC2)=O)C2CC2)CCc2nnnn2CC1 C1(NCC(N2CC3COCC3C2)=O)CCc2ccccc2C1 c1(CC(=O)NC(C)C(C)NC(c2cnc(C(F)F)s2)=O)cc(F)cc(Cl)c1 c1(C(N2CCC(C)(NC(C(C)CC3CC3)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 C1(NC(C=COCC)=O)CCN(C(=O)CC2CC(CC)=NO2)C1C C#CC1CC2CCC1N(C(C1C3CCN(C(=O)C=Cc4ccncn4)CC13)=O)C2 C12(C(=O)NCC3(CN(C(=O)CCCS(C)(=O)=O)C)CC3)CC3CC(C(=O)N1)C2C3 C1(OC)CC(CN(C)Cc2cn(C3CCCCC3O)nn2)N(C)C1 C12(NC(=O)NC(c3nnc4ccccn34)C)CCCC1CC(F)(F)CC2 CCCCC(C(=O)N1CCCC(C)C1CNC(C1CC(C)C1)=O)ON=C(C)C c1(-c2cc(C(=O)NC(C)CNC(C3(C)CC3C)=O)on2)cccc(F)c1 Cn1ccn2ncc(C(=O)NC3CCN(C(=O)CNC=O)C(c4ccccc4)C3)c12 CN1CCOCC1C(=O)NC1C=CCN(C(=O)CC2CC2)C1 N1(C(c2c(C)nns2)=O)CC2CCC(N=c3[nH]c4cc(Cl)cc(Cl)c4o3)C2C1 c1(NC(C2C(OC)C2)=O)nccn2ccnc12.C12CN(CCC1C(F)(F)F)C2=O c12ccc(nc1)N1CC(C1)OC2=O.N1(C(COCC(=O)NC)=O)CCOCC1 c1(C(=O)NC(C)CC(=O)N(C)CC2CC2)c(Cl)cccc1Br C1(CNC(C2C(=C)C2)=O)CC2CCC1N2C(=O)C1=C(C)OCC1 N1(C(C(C)(C)OC)=O)C2CCC1C(C)C(NC(c1cc(C)oc1C)=O)C2 C(=O)(CC(F)(F)C(F)F)NC1CN(C(C23CC(OC)C2C3)=O)C(C)CC1 C(CCNC(c1cccc(Cl)n1)=O)(C(C)C)NC(C1(C(=O)OC)CC1C)=O C1(CCNC(C2CC(SC)C2)=O)CC(F)(F)CN1C(C1CC2(C1)CC(C)C2)=O c1(CNCc2ccc(CCC)o2)cc2ccccc2[nH]1 CC(CCCCNC(C1CCCCN1S(C)(=O)=O)=O)NC(C1C(C)(C)C1(C)C)=O c1(OC)cncc(C(=O)NC(CNC(=O)C(F)C(C)(C)O)C2CC2)c1C c1(OCC)ccc(C(N2CCC(NC(C3CCN3C3CCCC3)=O)C2C)=O)cc1 c1(N2CCC(C)(OC(C)C)CC2)nc2c(c(=NCC3(C)CCCCC3)[nH]1)SCC2 c1(C(=O)NCC(O)CNC(c2coc(CC3CC3)n2)=O)csc([N+](=O)[O-])c1 C1(C(=O)NCC(C2CCC2)OCC)CNC(=O)CN1C(=O)C(=O)CC(C)C C(=O)(CCC1CCc2ccccc21)N1CCCCC(NC(c2onc(C)n2)=O)C1 C1(NC(c2nc(C)nn2C)=O)CN(C(=O)C(C#N)=CC2CC2)CCC1C C1(CC=C)(NC(C2CCCN2C=O)=O)CCCN(C(c2cc(COC)[nH]n2)=O)C1 c1(C(=O)NC2CC(C)N(C(c3ccc(C(F)F)cn3)=O)C2)cc2ccsc2s1 C(CC(C)C(=O)NC1CCC1NC(=O)CCN(C)CC)=CCC C1(CC(=O)OC)CN(CC(O)CCC2CC2)CC1O C1(NC(CCc2ccc(OCCC)cc2)=O)CCN(C(=O)CC(C)(C)O)CC1F c1(NCC(N2CCN(C(C3N(C(C)=O)CC3)=O)CC2)=O)ncsc1S(N)(=O)=O c1(C(=O)NC(CC(=O)NCCC(C)N2CCCC2)C(F)F)cc[nH]c2nccc1-2 C1(CNC(COCCCC)=O)CCN(C(c2nc(C3CC3)no2)=O)CC1C.OC N1(C(C=CCSC)=O)CCC(NC(=O)COc2ccnc(C(F)(F)F)c2)C(C)C1 O=S(=O)(c1ccc(SN2CC3CC3C2)cc1Cl)NCC1CCN(CCF)C1.C1(C)CC1 C1(CNC(C2(C=C)CCC2)=O)CN(C(=O)CC2CCSCC2)CCO1 C#CC1COCCN1C(=O)C(CC(C)C)NC(=O)OCC1CCCO1 CC(C)S(=O)(=O)c1ccc(C(=O)NCCC(C)NC(C2CC(C3CC3)C2)=O)cc1 n1(CCCC)nc(-c2ccc(C(C)(C)C)cc2)nc1C1CCCN(C(C)=O)C1 N1(C(C2=CC(C)C2)=O)CCN(C(c2cn(C3COC3)nn2)=O)CC(C)(C)C1 C1(C(C)(C)C)(NC(C2CC2F)=O)CCN(C(=O)CC2CCC3CC23)CC1 c1(NC(C(=O)NC(COC)C)(F)F)ccc(OCC)c(Cl)c1 C(=O)(C(CC(C)C)OC(c1cccc(C(F)F)c1F)=O)N1CCC(C(CC)C)C1 Cn1cc2c(n1)CC(C(N1CCC(F)(CNC(c3ccncc3)=O)C1)=O)CC2 c1(C(=O)NC(C(C)NC(c2ccc(C)cc2C)=O)C)cc2c(s1)CCCCC2 c1(C(C)C)cnc(O)c(C(N2CCC(C(C)NC(=O)CCCCC3CC3)C2)=O)c1 c1(C(=O)NC(c2nnnn2C2(C)CC2)CSC)cc2occc2n1C.N12CC(C1)C2 c1(C(CO)NCC(c2c(C)cccc2)O)ccc(F)cc1Cl C(N=c1[nH]c(Oc2ccc(OCCF)cc2)nc2ccsc12)C1CCN(C)CC1 c1(C(=O)OCC)cnc(NC(C2C3CN(C(c4ccsc4)=O)CC23)=O)c(Br)c1 c1(C(=O)NC2C(CNC(c3c(N)cc(F)cn3)=O)CCC2)noc2c1COCC2 c1(C(=O)NCCC2CCCN(C(CC(=C=C)C)=O)C2)cc(OC)cc2c1OCC2 C(CCC(=O)N1CCC(Cn2cc(-c3cccnc3)nn2)C1)N(C)C C(=O)(CCCN=[N+]=[N-])N1CC(C)C(NC(=O)CCc2cccnc2)C1.C(=O)(C)N C1(NC(C(C)C(N)=O)c2nnnn2CC2CCCO2)CC2(COCCO2)C1 C12(C(=O)NCC(=O)NC3CN(C(C4CC=CCC4)=O)C3)CC1CNC2=O N1(c2snc(C)n2)CCC(C(=O)NCC23CC(N(C)C)(CO2)C3)CC1 C1(C)(NC(CCN(c2c(OC)cccc2)C2CC2)=O)CC2=C(CNCC2(C)C)O1 n1(CC(=O)NC2C(NC(CC3CC(OCC)C3)=O)CCC2)cc([N+](=O)[O-])cn1 C1(NC(C(c2cccnc2)C)=O)(CNC(=O)CNC2(C)CC(F)C2)CCOCC1 N1(C(CCC(=O)OC)=O)CCC(CNC(C2CCC3CC3CC2)=O)C12CC2 N(C(=NCC1CC1)N1CCC(C)(OC)C1)CC(c1cccc(OCCOC)c1)O c1(CCNCC(N2CCc3ccccc32)C)cc(Cl)cc2c1OCC2 CCC(C)(CNC(c1cscc1Cl)=O)NC(=O)C(C)COC(C)(C)C C1(OC)CN(C(c2ccc(C(N)=O)o2)=O)CC1CO.c12ccnc(c1)N(C)C2=O C(=O)(C(C)C(=O)NC1CCCC1NC(C1(c2cccc(Br)c2)CC1)=O)OC Cc1ccnn1CC(=O)NC(C)CCCNC(c1cc(C2CC2)no1)=O n1(CC(=O)NC(C)CCNC(=O)C=Cc2cnc[nH]2)nc(C(F)F)cc1C(F)F c1(C(N(CCNC(=O)CC(c2ccccc2C)C)CC)=O)c(C)ncn(C)c1=O Nc1ccc(Cl)c(CNC(=O)NCc2cc(Cl)ccc2Br)c1 CC1=NOC(C(=O)NCC2(C(F)(F)F)CC2)C1.C12CC(C1)CNC2=O C1(NC(CC2(C)OCCO2)=O)CC(C(=O)N2CCOC(CCF)C2)=CC1O c1(CC(=O)NC2(C)CC(NC(C3CCCCCCC3)=O)C2)ccc2c(c1)COC2 C(CN=c1nc(N2CCC(NC(=O)CS(N)(=O)=O)C2)cc[nH]1)c1cc(C)no1 c1(C(N2CC(C)(C(=O)NC3CC3F)C2)=O)sccc1C#N C(C)(CCC(=O)NCC1CCCCC1C(=O)NCC(C)N=[N+]=[N-])OCC C1(CC(=O)NCCCOCCNC(CNC(=O)OC)=O)CCC2CC12 N1(c2nccc(C#N)n2)CC2(CCC(NC(=O)CN3CCCC3)C2)C1 Cc1ccc([N+](=O)[O-])cc1-c1c[nH]nc1-c1csc(-c2ccncc2C#N)c1 c1(C(=O)NCC2(F)CCCN(C(CSC)=O)CC2)n[nH]c2ccc(F)cc12 C(C(C(=O)N(C1CC1)Cc1ccccc1F)C(C)(C)C)NC(C(C)OCCOC)=O N1(C(C(C)Cc2ccco2)=O)CCN(CCc2nncn2C)CC1 CCCC(C(=O)NCC1(CC(N2CCC(CC)(CC)C2)=O)CC1)OCC n1(CC)ccc(C(=O)NCC(C2CC2)NC(=O)CN2CCCC2C)cc1=O CCCC(CC(C)C)C(=O)NCCNC(C1COCCO1)=O CC1C(C)N2CCN1C(=O)C(O)CCNC(=O)C2=O.C(C)(C)(C)OC(=O)N(C)C N1(C(C2CC(C#N)C2)=O)CC2CC1CN(C(c1coc(C3CCCCC3)n1)=O)C2 C1(C(CC)=O)CCCCC1O.C(CC(C)CCNCC)NC(=O)CCc1ccc(F)cc1 c1(CCCC)ccc(C(=O)OCc2cccc(COC)c2)cc1N N1(C(c2cn(C)c(O)n2)=O)CCCN(C(c2cccc(C(F)F)n2)=O)CC1 N1(C(CC(CN(C)C)O)=O)CCOCC(CNC(c2cn(C3CC3)cn2)=O)C1 c1(C(=O)NC2C(C(C)C)N(C(c3ccsc3)=O)CC2)nn(C)c(C(F)(F)F)c1Cl N1(c2cc(NCCOCC3CCOCC3)nc(CC)n2)CC2CS(=O)(=O)CC2C1 Cc1ccc(C(N2CCOC(CN(C)C(C3CCCC(C)(C)C3)=O)C2)=O)nc1C C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(=O)CN2CC(CO)C2)C1 c1(CCC)cccc(NC(=O)C(CC)NC(=O)C(CN(C)C)CC)c1 N1(C(CCCCC)=O)C(CNC(C2(COC)CCCCC2)=O)CC2COCC12 C1(C(N2CCC(NC(CCCc3nc(C)sc3)=O)C2)=O)CC2C=CCC(C1)C2 N1(Cc2c(-c3c(C4OCCC(C)C4)cccc3)cnn2C)CC2C(C1)C2(F)F N1(C(=O)CCCCc2ccc(Cl)cc2)CC2CN(C(C3CC(O)C3)=O)CC2C1 C(CCCCC(=O)N1CCC(C)(CC(=O)NCC)C1)OCC=CC C(C1CCc2ccccc21)NC(=NCc1ccc(SC)s1)NC1CC1 c1(C(N2C(CC(=O)NC(CCOC)COC)CCC2)=O)cc2n(n1)CCC2 Nc1ccc(C(N2CCC3C(NC(C4CCC(F)(F)C4)=O)C23)=O)cc1F C1(NC(C2N(C(CC)=O)CCCC2)=O)CC2CC1N(C(c1cc(C)cnn1)=O)C2 N1(C(C(C(C)(C)C)CNC(c2cc(CO)on2)=O)=O)CC2(C1)CC1(CCC1)C2 c1(C(C)C)cc(C(=O)NC2CC(NC(C3CC4(CCC4)C3)=O)C2)n(C)n1 Cc1ccc(CNC(C2(CCO)CC2)=O)c(-n2cc(C3CCCC(N)C3)nn2)c1 C1(C(N2CCC(NC(C3(NC(C)=O)CCC3)=O)C2)=O)CC2COCC(C1)C2(F)F C1(NC(c2ccc(COC)[nH]2)=O)CCC(CNC(=O)C(O)c2ccco2)CC1 C1(NC(c2nnc(C)s2)=O)CC(F)CN(C(=O)C(C)Sc2nnnn2C2CC2)C1 C1(OC)CCN(N(CC2CC2)CC2CC2)CC1 C#Cc1ccc(Oc2cccc(C(=O)N(C(=O)C(C)COC)C3CC3)c2)cc1 c1(C(N(C)CC2CCCN2C(c2cnc(C3CC3)s2)=O)=O)ccc(N)cc1[N+](=O)[O-] NC1CC2(C1)CC1(CC(F)(F)C1)C2C(=O)NNc1cccs1 C1(C(C)C)CN(C(c2cc(C3CC3)[nH]n2)=O)CCN1C(=O)CC1CCC(=O)C1C C1(CC(=O)OC)C(=O)NCCN1C(c1cc(F)ccc1C)C(=O)NCCCSC c1(C(N2CCOC(Cn3cc(-c4cccc(F)n4)nn3)C2)=O)cccc(F)c1F C1(C(=O)NC(C#C)C2CC2)CC2(CC2)CN1C(=O)C(C)NC(C)=O c1(CCC(=O)NC(CNC(CC2(N(C)C)CC2)=O)(C)C2CC2)cccnc1 c1(OC)cc(CN2CC3CCN(C(=O)Cc4ccsc4)C3C2)cc(CSC)c1O C(=O)(N=c1ccn(CCCO)[nH]1)C1CC(O)(CNC(CCC2C(C)(C)C2)=O)C1 CCC(O)C(=O)NCCCOCCNC(=O)CNC(=O)C(c1ccccc1)C C(CC1=CCCCC1)NC(C1CN(C(c2cnco2)=O)CC1F)=O c1(OC)c(F)cc(F)c(Cc2ncc(C(=O)NC(C3CCCO3)C)s2)c1F C1(C(N(C(CC)C)C)=O)CN(C(c2cn(CC)cn2)=O)CCC1(C)C Cc1nc(C)n(CCC(=O)NC2CCC(CCNC(=O)C=Cc3ccoc3)C2)n1 c1(NCCC)ccc(Cl)cc1C(=O)NC1CN(C(c2n[nH]cc2OC)=O)CC1O c1(C(=O)NC(CN(C(=O)C(C2CC2)OC)CC)C)cc[nH]c(=N)c1 CC1OC2CCC1(C(=O)NCC13CC1CN(C(=O)C(CN(C)C)NC(N)=O)C3)C2 C(=O)(C(C)(C)S(C)(=O)=O)Nc1cccc(NC(c2c(OC)ccc(CO)c2)=O)c1 O=S(=O)(c1ccc(N2CC3CC3C2)cc1Cl)NCc1cccc(Cl)c1 N1(C(CNC(C(C)(C)C)=O)=O)CC(CNC(=O)C2=CCC2)C2(CCC2)C1 CC1(C(=O)Nc2cc(F)ncc2F)CCCN(C(c2c(Br)cccc2Br)=O)C1 c1(C2C(C(=O)NC3(C)CC(NC(C4N(C)C(=O)OC4)=O)C3)C2)cccc(C#N)c1 C(=O)(CC(C(=O)NC1(CNC(=O)CC2CCOCC2)CCCCC1)NC(C)=O)OC c1(CCC)nc(C)c(C(=O)NC(C2CCCC2)CNC(c2c[nH]c(Br)c2)=O)o1 N1(C(c2cnc(C)nc2C)=O)CCC(NC(C2(C)CC2)=O)CC(O)C1 C1(NC(CCc2c(C)n[nH]c2C)=O)C2CC1CN(C(c1ccc(=O)n(C)c1)=O)C2 NC1C2CCCC1CC(C(N1CCOC(C3CC3)C1)=O)C2 C1(O)(C(C)CNC(=O)C=Cc2cncs2)CCN(C(=O)CC2CC(C)(C)CO2)C1 C1(CCC)CN(C(c2c(C)cccc2C)=O)CCN1C(=O)C(C1CCCC1)OC Cc1cc(C(N2CCC(O)(CNC(C3CCCC(=O)N3C)=O)C2)=O)cc(C)c1 Cc1nn(C)c(C)c1C1OCCC1NC(C1CC2(C1)CC(CNC(=O)CO)C2)=O C(C(C(=O)NCC1SCCS1)C(C)C)NC(c1cc(OCC)no1)=O Cc1cc(=NC2CN(C)C2CC2CC2)[nH]c(=NCc2ccc(C(F)(F)F)nc2)[nH]1 CC1CCCN(Cc2nc(CO)n(-c3cccnc3)n2)C1 C1(CNC(=O)NCc2ccc(CC)s2)CCCC2(CCOC2)O1 c1(C(N2CCCCC(NC(c3c(C)cc(F)s3)=O)C2)=O)cnn2c1OCC(F)C2 N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)CCc2nccs2)C(C)C1 N1(C(C2N(C(C)C)CCC2)=O)CCCC(F)(C(=O)NCCCC2C=NNC2=O)C1 CN1CCN(CC(N2CCN(C(=O)CC3CCCCC3O)CC2)=O)CC1 c1(C(NOCC(=O)NC(C)CCC2CCCC2)=O)ccccc1 c1(C(N2CCCC(N3CCN(C(CCC(=C)O)=O)CC3)C2)=O)cc(Cl)c(Cl)n1C C1(N(C(c2[nH]cc(C)c2C)=O)C)CN(C(=O)C(C(C)O)N(C)C)CCC1O C1(O)(CCOCCOC)CCN(N2CC(O)C3(CCOCC3)C2)CC1 C(C)(C(C)(C)NC(c1cnc(S)[nH]1)=O)NC(C(OC)OC)=O O=C(N=c1ccc(N2CCCCC2)n[nH]1)Nc1ccc(F)c(F)c1 N1(C(CC(C(C)C)C)=O)CC2CCC1CC2NC(=O)Cn1cnnc1O N1(C(C=CCOC)=O)CCN(C(c2ccc(COC)cn2)=O)CC1c1ncc[nH]1 CN(C1CC(C)(C)C1)N1CC(NC(=O)OC(C)(C)C)CC12CCC2 c1(CCC)cc(C(=O)NCC2CCN2C(=O)CSC2CCOC2=O)n(C)n1 C(=O)(C(C)(C)C(N)=O)NCC(CC(=O)N(C(C)COC)CC=C)C1CCC1 C1(N(C(C2C(=C)CC2)=O)C)CCC(NC(c2ccncc2N)=O)CC1 c1(C(=O)NCC2(O)CCN(C(CC3(C(=C)F)CCC3)=O)C2)nc[nH]c2ncnc1-2 N1(C(CCC(=O)NCC)=O)CCC(NC(=O)CN2C(=O)CCC2=O)CCC1 c1(OC)ccc(C(=O)NCCCN(CCO)C(C2OCCOC2C)=O)nc1Cl CC12CN(C(C3CCCC(=O)N3)=O)C(C(N3CCCCC(CO)C3)=O)(C1)C2 C(=O)(CCCCC(C)CC)N1CC(O)(CNC(COCCSC)=O)C1 N1(C(C)(C)C)CC(C(N2CCC3C(NC(=O)CCCn4cncn4)C23)=O)CC1=O c1(C(N2CCCC(CC(=O)NC3(CF)CCC3)C2)=O)cccn2nccc12 c1(N2CCOCC(C=O)C2)ccccc1S(C)=O.C(CN(CCOCC)CC)O CC1(C(=O)NCc2csc(C(=O)NC3(CCO)CCCC3)c2)CC=CC1 c1(C(=O)NC(CCCCNC(CC(=C)C)=O)C)cc(OC)ccc1F CC(C)CC(CNC(=O)CCCOC(C)C)C(=O)NCC(C)(F)C(C)C C1(C(N(CC(C)(O)C2CC2)C)=O)CCCN(C(C2(C#N)CCCC2)=O)CC1 CCC(C(=O)N1CCCC1CCC(=O)NCC1=NOC2COCC12)C(C)(C)CC C1(C(=O)NCc2c(C(=O)NC(CCN(CC)CC)C)n[nH]c2)CCCCN1C c1(CN2CC3(OCC(NC(c4ccc[nH]4)=O)C3)C2)n[nH]c2cc(Br)ccc12 Cc1cc(C#N)cc(C(=O)NNC(=S)NC(C(C)C)c2cccs2)n1 CC1(C(=O)NCC23CC2CN(C(C2(C#N)CC(=O)C2)=O)C3)CCCNC1=O C(=O)(CC(F)(F)C(F)F)N(C1CCN(C(C2CCCN2c2nccs2)=O)C1)CC C(=O)(C1=CCCC1)NC(C(=O)NCCCC(=C)Cl)C1CCCO1 N1(C(CCS(=O)(=O)N(C)C)=O)CCC(C)(C)C(NC(c2cc(F)cnc2O)=O)C1 C(CO)(C(=O)NOCC(=O)N(C)C)NC(c1onc(C)c1C)=O O=C1CCC(CC(N2CC3CC2C3C(=O)NCCN2CCC3CC23)=O)CC1 c1(C(=O)NC2CCN(C(C3CCC(=C)CC3)=O)CC2O)ccc(Br)c(C)c1C C(C1C(=O)N1C)N(C)C.C1(OC)CCN(C(C2(CS(C)(=O)=O)CC2)=O)C1.C(=O)NC=O C1(C)(NC(N(C(C(=O)OC)C)C)=O)C2CC3CC(C2)CC1C3 Cc1cccc(CCC(=O)N(C)CC2(O)CN(C(c3cnc(C(F)F)s3)=O)C2)c1 CC1(NC(=O)Cc2csc(Cl)n2)CC(NC(C2CC2Cl)=O)C1 Cc1cc(NC2CC(F)(F)C2)ncc1S(=O)(=O)NCC1CCOC(C)C1 CCC(CC)C(F)C(=O)NCCOCCCN(C)C(C1CCN(C(C)=O)C1)=O CCC(C)CC(C(=O)N1CCCC(CC)(CO)C1)NC(=O)C(F)(F)F C1(NC(COCC=C)=O)CCC2(CCCN(C(c3cocc3Br)=O)C2)C1 N1(CC(=O)NC2CCC2c2ccccn2)C(=O)C2CC=CCC2C1=O C#CCCC(N)C(=O)N1CC(C(=O)O)CC1(C)C Cc1ccc2cccnc2c1C(=O)NCCC(C)(C)NC(=O)CC1CCCC1C C(=O)(C1CCc2ccc(OC)cc21)NCCCN(C(C1C(=C)C1)=O)C Cc1ccnc(F)c1NC(C1CC12CCN(C(=O)C(c1cccc(Br)c1)O)C2)=O C1(C(N(CC)CC2CC2)=O)N(C(C2CCC(O)CC2)=O)CC12CCCC2 c1(C(=O)NCC(CNC(C(C)(F)F)=O)CO)ccc(N2CC(F)CC2=O)cc1 C1(C(=O)NC(CCOC)CNC(C2(C)CC2C)=O)CC2(CCCC2)C1 C(CC(C)C)(C(=O)Nc1ccc(C(n2cc(CC(O)C(C)C)nn2)=O)o1)OC C1(CCC)CN(C(=O)C=CC=C(Cl)Cl)CCN1C(=O)CC1CCCC(C)(C)C1 c1(C(=O)NCC(CNC(C2CCC(C)O2)=O)(C)C)ccc(OC(C)(C)C)cc1 CC1C(C(=O)NC(c2ccn(C)n2)C)CCN1C(=O)C(C1CCCCC1)O C1(NC(c2cc(OC)cc(Cl)c2)=O)CC2(CCN(C(C3CCC3(C)C)=O)C2)C1 C1(N(C(C=NOC)=O)C)CN(C(c2ccn(-c3cccc(C)c3)n2)=O)CC1(C)C CC(C)CCC(C(=O)NC1CCN(C)C1(C)C)NC(=O)C(C)OC(C)(C)C c1(C(N2CC(NC(c3ccc(Cl)c4occc34)=O)C2)=O)ccc2ccnn2c1 N1(CCOCC)CCN(C(C2CCCC(Nc3ccc(CC)cn3)C2)=O)CC1 Cc1ccc(Br)c(F)c1C(=O)NC1(C)CCOC1C1CC1 C#Cc1ccc(C(=O)N(C(CNC(C2(CC(F)(F)F)CC2)=O)CC)CC)c(F)c1 N1(C(c2cnc(C3CC3C)s2)C(=O)NCCCC(=O)OC)CCNC(=O)C1(C)C C1(C(N2CSCC2C(=O)NCC(C)C(F)F)=O)(OC)CCC(C)C1 c1(N2CCCC(C(=O)NCc3c(C)c(Br)ccc3)C2)ncnc2cc(I)sc12 c1(C(N2CC(NC(CCC#C)=O)C(C=C)C2)=O)cc(Br)ccc1[N+](=O)[O-] c1(OC)cnc(F)c(C(=O)NCC2CCCN(CCOC3CCCC3)C2)c1 c1(CC(=O)N(CC)CC2CCN(C(=O)CCN(C)C)CC2)cccc(C)c1Cl c1(OC)ncc(CN2CCOCC(C(=O)N(C)CC3CCCCCC3)C2)cc1C N1(C(CNC(C)=O)=O)CCCC(O)(CNC(C2CC(C3CCC3)C2)=O)CC1 N(C(=NCc1ccccc1)N1CCC(C(=O)Nc2cc(C)ccn2)C1)C(C=C)C c1(C(N(C(CNC(CCCNC(C)=O)=O)C)C)=O)ccc2ncnc(O)c2c1 C(CCC(C)CC(=O)N1CC2C(C1)N2Cc1c(C)noc1C)=C(C)C CCCC(CCC)C(=O)NC1(CN(C)C(c2onc(Br)c2C)=O)CC1 c1(C(=O)OCC)cc(C(=O)NCC(O)CNC(C2COC(=O)N2)=O)n(C)n1 CC12COCC1CN(C(C1N(C(=O)C3=NNC(=O)C3)CC13CCCC3)=O)C2 c1(C(=O)NCCC(C)N(C)C(C2CNC(=O)N2)=O)ccc2c(n1)CCC2=O CC(C)C(O)CC(=O)NC(Cc1cn[nH]c1)C(=O)NCCN1CCNC1=O Cc1cc(C(N2CC3CC3(CNC(=O)CCCC3CC3)C2)=O)c(C(F)(F)F)o1 c1(C(=O)NC2CC(NC(=O)CC34CCCN3CCC4)C2)cc([N+](=O)[O-])ccc1F N1(C(c2c(C)nn[nH]2)=O)CCC(C)N(C(c2cc(Cl)cnc2O)=O)CC1 C(CC(C)(O)CN1CCC(c2cccnc2)C1)OC C(C(O)C(=O)N1CCCC1C(C)(C)CNC(c1cc(Br)n[nH]1)=O)N(C)C c1(C(N2CCOCC(CNC(C3C(C=C)C3)=O)C2)=O)cc(F)c(C(F)F)c(F)c1 Cc1ccc(NC(=O)CN(C2CC3CCC2N3C)C)cc1C C#Cc1ccc(NC(=O)C(=O)Nc2cnn(CCN3CCCCC3)c2)cn1 C(=O)(C1=CCC2CCC1N2C(C1(C)CCC(F)(F)CC1)=O)OC(C)(C)C N1(C(Cc2ccc(OC)c(F)c2)=O)CC(CNC(C2(C)CCC2)=O)CC12CCC2 N1(C(C2C=CCC(C(=O)OC)C2)=O)CCC(C)(n2ccnc2)CC1 Cc1ccc(F)cc1CN(C(=O)CC1CC1CNC(=O)CC1CCCCC1O)C N1(C(CCN(CC#C)C(C2CC2C(C)(C)C)=O)=O)CC(F)(F)C1 c1(C(c2n(C)nnn2)Nc2nccs2)ccccc1[N+](=O)[O-] CCC(C)(CNC(=NC)NCC1(C#N)CCC1)OC c1(CC(C)C(=O)NC2CC(NC(=O)Cc3ccco3)CC2O)cccc(Cl)c1 C1(CNC(C2(n3cc(C(C)(C)O)nn3)CC2)=O)C=CCN1C(=O)OC(C)(C)C N1(C(=O)CNc2nccs2)C2CCC1CC(NC(C1(O)CCOC1)=O)C2 c1(C(=O)NC)cscn1.c1(CNC(C2(C(C)C)CCC2)=O)cc(CC2CC2)n[nH]1 N1(C(c2cccc(C3CC3)c2)C(=O)NCC=C)CCCC(C)C1CC N1(C(C)=O)CCOCC1c1cn(-c2cc(NC)oc2C)nn1 c1(C(N2C(CNC(C3C(C)C3(F)F)=O)CC2)=O)nccc2[nH]ccc12 C1(NC(CC2(C(C)(F)F)CC2)=O)(CO)CN(C(=O)Cn2nnc(C3CC3)n2)C1 c1(OC)cccc(C(CNC(C2CC3CC2C3)=O)NC(=O)CCC(F)F)c1 c1(C(C)NC(=O)NCc2cc(N(C)CCO)ccn2)cc(F)c(F)c(F)c1 C(=O)(C#CC1CCCCC1)NC1CCC(NC(c2ccc(C)c(Cl)c2F)=O)C1 c1(OC)ccc(CCN)cc1C(=O)OC.c12cn(nn1)CCNC(=O)CC(=O)NC2 n1(CC(=O)NC(C)(CNC(c2nccnc2O)=O)C2CC2)cnc([N+](=O)[O-])n1 C(c1ccc(F)cc1F)=CC(=O)NC(C1CC(NC(=O)CCN2CCCC2)C1)C c1(C(N(CCN(C(=O)C(c2cccs2)C)CC)CC)=O)cn(CC(N)=O)nn1 CC1CCN(C(=O)COCc2cccnc2)CCN1C(C1CC(C(C)(C)C)C1)=O C(=O)(C(C)CCCC)NC(CC(=O)N(C(CCSC)C)C)COC c1(C(N2CC(NC(c3ccn(CCN(C)C)n3)=O)(CO)C2)=O)c(F)cccc1Cl c1(C(C(=O)NCCN(C)C(C23CCCC2C3(F)F)=O)(C)C)ccc(F)c(Cl)c1F C(CCS(C)=O)(C(=O)NC1CCC(NC(c2ocnc2C2CC2)=O)CC1)N(C)C C1(CNC(CC(=C)C)=O)CC(C(C)C)CCN1C(c1cnccc1OC)=O Cc1ccc(F)cc1CC(N1CCCCC(N(C(=O)C2=NOCC2)C)C1)=O N1(C(CC=CC=C)=O)CCCCC1C1(NC(c2cc(C)co2)=O)CC1 c1(C(=O)OC)ccc(C=CC(N2CCCC2CN(C)C(C2(CCO)CC2)=O)=O)o1 C1(CNC(c2c(F)ncc(C)c2)=O)CC2(CCC2)CN1C(=O)C(C#N)=CC1CC1 N1(C(c2c(C)[nH]c3ccccc32)=O)CCCC(C2CN(C(C3C4CC5C(C4)C35)=O)C2)C1 c1(C(=O)NC(Cn2cc(C=CC)nn2)C)cnc(C)c(Br)c1Cl C1(N(C(=O)Cc2ncc(C)s2)CC)CCN(C(C2(C)CC2(C)C)=O)CC1 C1(C)(C(=O)NC(CC(=O)NC)C)CCN(C(C2CC2(F)F)=O)CC1 Nc1c(C(N2CCCCC2CNC(=O)C(F)(F)C(O)C2CC2)=O)ccnc1Cl CC1=C(C(=O)NCC2CCOC2C(=O)NCC2CC2c2ccoc2)CC1 c1(CC(=O)NCCN(CCCC)CCOC)c[nH]c2ccc(C)cc12 N1(C(CC(=O)NCC#C)=O)CCN(C(C2(c3ccc(F)cc3)CC2)=O)CC(O)C1 N1(C(C2CC(C)(CC)C2)=O)CCC(NC(c2cccc(COC)c2F)=O)C1(C)C C1(C(=O)NC2(CCCC)CC2)C(C)CCN1C(c1cncc(NC)n1)=O CCC(O)C(F)(F)C(=O)NC1CC(NC(=O)CN2CC(C)(C)C2)C(O)C1 C1(C)(CNC(c2cnc(CC)nc2O)=O)CC(F)(F)CN1C(c1cn(C)cn1)=O Nc1ccc(Cl)c(C(N2CCC(CCNC(C3CC(O)CN3C)=O)C2)=O)c1 c1(COCC(=O)NC(CC=C)CNC(=O)Cc2cc(OC)no2)ccccc1Cl C(=O)(CC(C)(C)O)NCC1N(C(c2c(CC)[nH]cc2)=O)CC1 c1(C(N2CCC(CN(C(=O)Cn3cccnc3=O)C)C2)=O)c(O)ccc(F)c1F c1(CCCC(=O)NCC2CN(C(C3OCCCO3)=O)CCO2)cc(F)ccc1F C1(NC(c2c(C)nc(COC)s2)=O)CC(F)CN(C(c2cc(C)ncc2C)=O)C1 C=CCC(CNC(c1[nH]ccc1C1CC1)=O)C(=O)N1CCC(CC)C1 C12(C(=O)NC(C3CCOC3)CNC(=O)CSc3ccccn3)CC1CNC2=O CN(CCCC(=O)NC(c1ccc(F)cc1)CNC(=O)Cn1cncn1)N=O c1(C(C)C)cc(C(=O)NCC2CCCCN2C(=O)Cc2cncs2)ccc1F C1(NC(=O)CC2(O)CCCCC2)CCCN(C(=O)CCc2ccoc2)CC1F C1(NC(c2ccc(C)s2)=O)CCCCCC1C(N1CCC1CN=[N+]=[N-])=O CCC(CCC(=O)NCC1CCSC1)NC(=O)C(C)(C)O c1(CNCCCN2CCCC(OC)C2)cc(C)c(Br)c(Cl)c1 Nc1ccc(F)cc1C(N1CC2CC(CNC(c3ncccc3CO)=O)C2C1)=O C(=O)(C1Cc2ccccc21)NC1CCN(C(c2ccc(CSCC)o2)=O)CC1F N1(C(CCn2ncc(C)c2)=O)CCCOC(CNC(c2ccc(Cl)c(C)c2)=O)C1 C1(NC(C(c2c(C)nn(C)c2)C)=O)CCN(C(C2CNC(=O)O2)=O)CCC1CO Cc1ccnn1C(C)C(=O)NC(C)(C)CNC(=O)C(C)Cc1ccccn1 C(=O)(C(F)CC(C)(C)NC(C1CCCSC1C)=O)NC1CC(C)(CC)C1 CCCCC(C(=O)NC(CCOC)C(N)=O)NC(c1cc(C2CC2)no1)=O c12cccc3c(c[nH]c13)C(=O)OC2.c1(OCC(=O)NC)ccccc1C N1(C(CC)=O)CCC2(CCCN2C(=O)C(C)CC(=O)c2ccc(F)cc2)C1 c1(C(=O)NCC2CC(OC)CN2C(C2COCCOC2)=O)cc(N)ccc1Cl c1(CC=C)cc(C(=O)NCC(C)NC(=O)Cc2nnc(O)s2)cc(OC)c1OC c1(CC(=O)NCCC(C)NC(CCn2ccc(C)n2)=O)nn(C)cc1[N+](=O)[O-] c1(C(=O)NC(C(C)C)CNC(C2CCOC2C)=O)ccn(CCO)c(=O)c1 C1(CC)CN(C(c2cccc(C3(C#N)CC3)c2)=O)CCN1C(c1ccc(C)o1)=O C(=O)(C(C(C)C)C(C)C)NC1C2CN(C(c3ccc(CCC)cc3)=O)C1CC2 C1(CNC(C2CCCOCC2)=O)CN(C(C2CCCCS2)=O)CCC12CCOC2 CC(CC(C)(C)CO)NC(=O)CC1N(C(c2nc(=N)cc[nH]2)=O)CCC1(C)C C#CCC(CC(F)F)C(=O)N1CCN(C(c2sc(O)nc2C)=O)CC12CC2 O=C(C1=CS(=O)(=O)c2ccccc21)NCC12CC(c3ccccc3)(CO1)C2 C(=O)(C(C(C)(F)F)c1ccccc1)NCCN(C(=O)C=CCN(C)C)CCOC C1(C(N(CCCOCCNC(C2(c3nc[nH]n3)CC2)=O)C)=O)CC12CC(O)C2 c1(C(C)NC(c2cc(Br)c(F)cc2F)C)cc(F)c(N)c(F)c1 N1(C(=O)CC2CC=CCC2)CC2CCCC2(Nc2ncncc2Cl)C1 N1(C(C(c2cccc(C)c2)C)=O)CC(=O)NC2CN(C(c3cnsn3)=O)CCC12 c1(C(=O)NCCC2N(C(C=C(C)C(C)(C)C)=O)CCC2)cc(C)c(Cl)cc1F N=c1[nH]cc2c(c1C(N1CCC3(CCC3NC(=O)CC3CCC3)CC1)=O)CCC2 N1(C(Cc2nnc(C)o2)=O)CC2(C)CN(C(C3CC3C)=O)CC2(C)C1 C(=O)(C(C)(C)CCC#N)N1CCC(C(=O)NCC2CCCC(C)O2)C(O)C1 Cc1onc(Cl)c1C(=O)NC1CN(C(C2SCCS2)=O)CC1CC1CC1 CC(C(=O)NC1CCN1CCCNC(=O)CNC(=O)NC1CC1)C1CCCC1 C1(NC(C=CC)=O)CN(C(c2cnn(-c3nccs3)c2)=O)C2(CCOC2)C1 c1(CC(=O)NCC2(C)CCN(C(=O)CN3CC=CC3)C2)cccc2ccccc12 c1(CCC(=O)NCC(C(C)(C)C)NC(C(COCC)C)=O)cc(F)cc(F)c1 C12(C(N(CCOC)CCO)=O)CCC(CN(C(=O)C(=O)C(C)C)C1)C2 C1(NC(Cn2ncc(C)c2)=O)C2CCCN(c3ncnc(O)c3Br)C2C1(C)C N1(C(c2nc(C)oc2C)=O)CC2CCC1CN2C(=O)C(C(C)(C)C)n1ccnn1 c1(C(N2CCC(C(N3C(C)(C(=O)OC)CCC3)=O)C2)=O)ccc(F)cc1C c1(C2CC(=O)NC2)cccc(CNCc2cnn(C3CCC3)c2)c1 c1(C(N2CCC3CN(C(C4CCSC4)=O)C3C2)=O)cc2nccc(Cl)c2s1 c1(NC(C2N(Cc3ccc(C#C)s3)CCC2)=O)cnc(Cl)c(C#N)c1 C(C(C)C(C)C(=O)NCC1(NC(c2ncoc2C2CCC2)=O)CC1)OC C(=O)(C1=COCCO1)NCC12C(CN(C(C(c3n(C)ccc3)=O)=O)C1)C2 CCC(CC)(CCNC(=O)CCc1cncnc1)NC(c1nccc(N)c1Cl)=O C(C)(C(O)C(=O)NC(C)(C)CCNC(c1cccc(N(C)C)c1)=O)SC N1(NC(C2CCC(NC(C3CC(C#C)(O)C3)=O)CC2)=O)CC2(C1)CC1(CCC1)C2 C(C(C(=O)NCCCSCN1CCOCC1)NC(=O)Cc1cnns1)OCC N1(C(c2[n+]([O-])ccc(OC)c2)=O)CCCN(C(c2ccc(C)s2)=O)C(C)C1 c1(CCC(=O)NCC(=O)NC(CNC(C(C)C)=O)(C)C)ccccc1 c1(C(=O)NCC(CNC(=O)CCc2cn[nH]c2)OC)cnc(S)n1C1CC1 CC(F)(F)C(F)C(=O)NC1CC(NC(c2cc(Br)cnc2O)=O)C1 c1(OCCN2CCC(c3ccc(C#C)s3)C(O)C2)c[nH]c2cc(OC)ccc12 N1(C(CN2CCC(C)(C)C2)=O)CC2(C1)CN(C(C1CC3CCC13)=O)C2 N1(C(c2nc(COC)sc2)=O)CCCC(NC(C2(C)CCCS2)=O)CCC1 c1(N(C)C)ccc(C(=O)N(C2CCN(C(=O)CC3C(C)(C)C3(C)C)C2)C)nn1 N1(C(CS(=O)(=O)NC)=O)CCCC12CCN(Cc1ccc(O)cc1C)CC2 C1(C(N2CCC(C)CC2)=O)CC(N=c2c([N+](=O)[O-])c[nH]c3c(Cl)cccc23)C1 c1(CN2C(C(=O)NC3CN4CCC3CC4)CC3CC32)c[nH]c2cccc(Cl)c12 c1(C2CC(C(=O)NC(C)Cn3cc(CC4(O)COC4)nn3)C2)ccc(Cl)c(Cl)c1 N1(C(C=CCC(C)(C)NC(=O)Cn2[nH]cnc2=N)=O)CCCC2(C=CCO2)C1 C=CCC(CC(F)F)C(=O)N1CC(NC(c2cc(F)cc(Br)c2C)=O)C1 C1(CNC(C(CO)N(C)C)=O)CC2(CCC2)CN1C(c1cc(O)nc(O)c1)=O C1(c2cn(-c3n(C)nnc3)nn2)CC12CCN(C(=O)CCP(C)(C)=O)CC2 c1(C(=O)NC2CN(C(c3c(N)ccc(CC)c3)=O)C2)nccc2ncncc12 c1(N2CC(C)OCCC2)ccc([N+](=O)[O-])cc1[N+](=O)[O-].N1(C(C=C)=O)CCNCC1 C(C)(CCCCC)(C(=O)NCCN(C)CCF)NC(C1C(=C)C1)=O N1(C(C23OCC(CC)(C2)C3)=O)CCN(C)C(CNC(=O)CCSCC(C)C)C1 C(C)(CNC(=O)C(F)OC(F)(F)F)(CC(C)C)NC(c1c(OC)n(C)nc1)=O c1(C(N2CC(C(C)Nc3ncc([N+](=O)[O-])cn3)C2)=O)ccc2oc(=O)oc2c1 c1(C(=O)NC(CNC(CSCC=C)=O)(C)C)cc(C)ccc1F c1(C(=O)NCCCN(C)C(c2ccnc(OCCO)c2)=O)c(F)cncc1Br C(=O)(CC(CC)N(C)C(C1CC=CCC1)=O)NCc1cc(CC)no1 c1(CC)cnoc1C(=O)NC(CO)C(=O)NC(C1CCC1)C C1(C(=O)NCCCN(C)C(C2CC3(C2)CC3F)=O)(C(F)F)CCCCC1 C1(CNC(c2ccc(COC)cc2)=O)CN(C(=O)C(F)(F)C(F)F)CC12CC2 C1(O)(CC(C2CCOCC2CO)=O)CCOCC1.C12CCCC1CC(=O)NC2=O C1(N(C(C(C)Cn2ccnc2)=O)C)CCCN(C(=O)CC(C)(O)C2CC2)C1 Cc1cc(CO)oc1C(=O)NCCC1CCN(C(=O)CC2COCCN2C)C1 N1(C(CC(CC)O)=O)CCC2(CCCN2C(c2cc(CO)oc2C)=O)C1 N1(C(CC2CCCC(C)C2)=O)CCCC2(CNC(=O)C=CBr)CCCC12 C(=O)(C(C)C(F)(F)F)N(CCCN(C(=O)C1CC1)CC)C.C1(C(C)O)CC(F)C(=O)N1 C12(NC(CS(=O)(=O)NC)=O)CCC(CN(C(C34CCCC3C4(F)F)=O)C1)C2 O=C(C1CSc2ccccc21)NCC=CCNC(C1(c2ccccc2)CC(O)C1)=O C1(C(=O)NCC=C(C(=O)NC(CCC)CO)C)(CO)CC(C)(C)C1 C1(CNC2CC3(C2)CC3F)CN(C(c2ccc(C(=O)NC)cc2)=O)CC(C)(C)O1 c1(C(=O)NC(CN(C(C(C(C)C)O)=O)C)C)nc2ncc(Br)cc2[nH]1 C1(NC(c2c(C#C)cnn2C)=O)CN(C(C2CCC(N(C)C)C2)=O)CCC1(C)C S(=O)(=O)(CC(=O)NCC1CCCN1C(c1cnn(CC2CCOC2)c1)=O)NC c1(Oc2ccc(-c3nn(CCOC)c(CC(=O)OC)n3)cn2)ccc(C)cc1Cl c1(C(=O)NCC2N(C(C3N(CC)CC3)=O)CC2)cc(N)cnc1C c1(NC(=O)CC(=O)N)cccc2ccccc12.C1(C(C)N)CC1CNC(=O)C1CC1 CCCCCCCCS(=O)(=O)N1CCCC1CS(N)(=O)=O O=C1CCN(C(c2ncccn2)=O)C(C(N2CC(F)CC2C)=O)C1 CC1CCOCC1C(=O)NCc1cccc(NC(=O)Cn2cccnc2=O)c1 C1(n2cccn2)(C(=O)NCCN(C(C)C(=O)Nc2ccccc2)CC)CCCC1 C1(COC)CN(C(=O)CSCC(F)F)CCN1C(C1CCN(CC(F)F)CC1)=O N1(C(C2CN(C(CCOC)=O)CC2(C)C)=O)CCNC(=O)CC1C CC1C(C)N(C(=O)Cc2cncnc2)CCN1C(c1cnn(C)c1N)=O CC(C(C)C(=O)NC(C)(C)CN(C)C(C12CC(N=[N+]=[N-])C1C2)=O)C(C)(C)C C1(CNC(C23CC(C(=O)Nc4cccc(F)n4)(C2)C3)=O)CCC2CC2C1 N1(C(C2(C)CCC(=O)N2)=O)CC2CCC(C1)N2C(c1ccn(CCF)n1)=O N1(c2cc(NCC3(CSC)CCC3)ncn2)CCC(CO)C(C)C1 c1(C(=O)NC(C(C)C)C(C)NC(C2C3CCC2CC3)=O)ccc2ccoc2c1 Cn1ccc(C(=O)NCC2CN(C(=O)CC3(C)CC3(Cl)Cl)C2)cc1=O c1(C(=O)NC(CC)CN(C(=O)CC(=O)OC)C)cc(OC)c2c(c1)CCO2 N1(C(c2cc(Br)cs2)=O)CCOCC1Cc1cn(CC2(F)CCOC2)nn1 C1(CCC(=O)Nc2c(C(=O)OC)n[nH]c2)CN(C(=O)C=CCBr)CCO1 c1(C(=O)NCCC(=O)NC(CC)C)cc2c(cc1Br)OCCO2 CC(O)C(C(N)=O)NC(=O)C(CN(C)C)NC(=O)CNc1cccnc1 c1(C(=O)NC2C(NC(C3C(C(C)=O)C3)=O)CCC2)cccc(C(C)(F)F)c1 C(N=c1nc(N2CCc3nc(Br)sc3C2)c2[nH]ccc2[nH]1)C1(OCC)CCCC1 CCC(C)CC(C)C(=O)N1CCC(C)(NC(=O)Cc2cccc3ccoc23)CC1 N1(C(C(N2CCCCC2=O)C)=O)C2CCC1CN(C(C1CC1(C)C)=O)CC2 CCCC(O)C(CO)NC(C1C(CC)CCN1C(=O)CC1(OCC)CC1)=O N1(C(c2c(CC)nccc2)=O)C2CCC1CN(C(=O)CCC(CC)OC)CC2 c1(NC(C23N(C(CC(C(C)C)C)=O)CCC2C3)=O)ccc2cncn2c1 C1(CCNC(CN(C)C2CC2)=O)CCCCN1C(C1CCCCC1O)=O Cc1cc(NC2CN(C(=O)C=Cc3ccsc3)CC23CCC3)n2ncnc2n1 N12CC(C3(CCC3)C1)C1C(C)(C1)NC2=O.CC(C)(C)OCC(O)C1(C)N=N1 S(=O)(=O)(c1cnn2ccc(NC3CCn4nccc4C3)nc12)NC(C)(C)C C(CSc1ccccn1)(C(=O)NCC1CCN1C(=O)CCF)NC(C)=O C(=O)(C1=C(F)CN(C(C2CS(=O)(=O)C2)=O)CC1)NC1C(C#N)CCCC1 N1(C(C2C(C#C)C2)=O)CCC(C)(CNC(c2ccc(-n3cccn3)nc2)=O)CC1 C(=O)(CC(C)(C)CNC(C12CCCN1CCC2)=O)NCCCSC N1(C(C2CCC(=O)C2)=O)CC2CCC1C(CNC(C1C(C3CC3)C1(F)F)=O)C2 C1(C(=O)NC(CO)CCC2CC2)CN(C(=O)C=Cc2ccoc2)CC1F c1(C(=O)NC2(C)CC(NC(c3csc(C(F)(F)F)c3)=O)C2)cc2n(n1)CCCC2 C1(C)(NC(CCCn2c(C)ncc2)=O)CCCN(C(=O)CCCN(C)C)C1 c1(C(C)=O)ccccc1C(=O)NC1CCCC1NC(=O)C(C)(C)c1ccnn1C n1(CC)nc(C)c(CNC(N2CCC2CSc2ccccc2)=O)c1C c1(OC)cc(NC(C2CCCN(C(c3cccc(Cl)c3OC)=O)C2)=O)c(Br)cn1 C(CC(C(=O)NC(C)CN(C)C(c1sc(C(C)(C)C)nc1C)=O)OC)OC CC1CC(C(C)(C)C)CN(C(=O)C=CC(=O)N(C)C)C1.C12CC=CC(C1)C(=O)N2 N1(C(c2ccc(NC(C)C)nc2)=O)CCC2(C1)CN(C(=O)Cc1ccns1)C2 CC1(C)COCCC1C(=O)NCC1CC2CN(C(=O)Cc3ccc(O)cc3)CC12 O=C(C1=CS(=O)(=O)CCC1)NCC1CCN(C(c2cncc(F)c2)=O)CC1(F)F CCC(CC)(CC)C(=O)N1CCC(C)(NC(c2ccc3nc[nH]c3n2)=O)C1 N1(C(c2scc(C)n2)=O)CCN(C(=O)Cc2cncc(O)c2)C(C(F)(F)F)C1 C1(O)(C(=O)NCC2CC(C(=O)NC3C4(CC(OCC)C4)C3)C2)CCOC1(C)C N1(C(c2n[nH]c(C)c2Br)C(=O)NCCOCC2CC2)CC(C)NC(=O)C12CC2 C(C(C)C(F)C(=O)NCCn1cnnc1)NC(CC(C)C)=O OCC(CO)(CO)C(O)CN1CCC(CCO)C1 CC1CN(C(=O)CC2(C(F)F)CC2)CC1CNC(=O)CCCOc1ccccc1 N#Cc1c[nH]c(C(=O)NC2CCC(NC(=O)CCC3CCCCC3)C2)c1 C1(NC(Cc2cc(C)c(F)cc2)=O)CC2CC(NC(=O)CC3(C)CC3)CC2C1 Cc1cccnc1CC(=O)NCCCNC(=O)C(C)n1cccn1 c1(C(=O)NCC2N(C(C3(CCCC)CC3)=O)CCC2)cccc(CCCCO)c1 c1(OC)ccc(N2CC(C(N3CC(CNC(=O)C(F)C4CC4)C3)=O)CC2=O)cc1 C1(CC(C)C)CS(=O)(=O)N1N(Cc1ccccc1)C(C)c1ccncc1 c1(OC)ccnc(C(=O)NCC2CCC(C)CN2C(=O)CC2(OC)CCC2)c1C c1(CN(CC(C)CO)C(=O)OCc2cscn2)ccccc1 C1(SC)CN(C(=O)CCOCc2ccccc2)CC1NC(=O)CN1CCCCC1 N1(C(c2ccccn2)=O)CCCCC(NC(c2cn(CC(=O)OCC)nn2)=O)C1 C1(C)(C(N(CC(C)NC(C2(C3CCCO3)CCOCC2)=O)C)=O)CCCCO1 CC1CC=CCC1C(=O)NCC(O)CNC(=O)CCNC(c1ccccc1F)=O N1(CC(=O)N(C(C)CN(C)C(c2ccc[nH]2)=O)C)CSCC1=O N1(C(C(CC=C)C)=O)CCC2(CC1)CC(NC(=O)CCNC(=O)COC)CCO2 C#CCC(CC(=O)N(CC(C)OC)C(C)C)NC(c1cnnc(O)c1)=O c1(C(=O)N)nccc2ccncc12.N1(CCn2cncn2)CCN(CC2CC2)CC1 C1(CNC(C2(COC)CCCO2)=O)CN(C(C)=O)CC1O.c12n[nH]cc1NC2=O C1(C)(C(=O)NCCCCNC(c2ncn(C(C)(C)C)n2)=O)CCSCC1 N1(C(C2CC2(F)F)=O)C2CCC1CC(NC(C1(c3ccccn3)CC1)=O)C2 C1(CC(=O)NC(CN(C(CC(=C)Br)=O)C)C)CCN(C)CC1 c1(C(=O)O)cc(C(=O)NCC2(Sc3ccccc3)COC2)n2ccsc12 N1(C(CN(C2CCC2)C)=O)CC2CC2(CNC(C2COCCN2C(C)=O)=O)C1 c1(SC)nccc(=NCC2CN(C(C3COCCO3)=O)CC23COC3)[nH]1 c1(C(=O)NCC2C(NC(C3NC(=O)CC(C)C3)=O)C2)ccc2c(c1)nnn2C CN1CC2(CCN(C(C3CC(F)CN3Cc3ncc(Br)cc3Cl)=O)CC2)C1 c1(C(C(C)N(C)CC2CCN(C)C2=O)=O)cccc2ccccc12 N1(C(c2cnn(C(C)C)c2C2CC2)=O)CCC(CNC(C2CC2(C)Br)=O)C(C)C1 N1(C(C=CCOC)=O)CC2(CC(NC(c3snnc3C)=O)C2)C1 C#Cc1ccccc1CN1CC(CC)OC(C)C1 c1(NCC(C(C)(C)C)NC(c2ccc(CC)s2)=O)nc(O)c2c[nH]nc2n1 CC(CN=c1nc(N(C)Cc2ccc(F)c(Br)c2)c2cccc(F)c2[nH]1)C(F)F N1(C(C(=Cc2cccs2)C)=O)CCC2(CCCC2NC(=O)CCC(C)(C)C)C1 c1(C(N2C(CCNC(c3cncc(N)c3)=O)COCC2)=O)cccc(=S)n1O N1(C(c2c(F)ccc(N)c2)=O)CCC(NC(=O)CC2=CCCC2)C(CO)CC1 c1(C(=O)NC2C(C)CN(C(=O)CC3(CO)CCCCC3)C2)ccc(N)cc1F c1(C2N(Cc3c(OC)cccc3Cl)CC3CN3C2)ncc2cc(Br)cnc2n1 Cc1nnc(CSc2ccccc2C(=O)NNC(=O)Cc2ccsc2)nc1C C1(CCNC(c2c(C)ocn2)=O)CN(C(=O)CCCc2nccs2)CCCO1 NS(=O)(=O)CC(=O)NC1CC(NC(=O)CC2CCCOCC2)C1 N1(C(C2CC(n3cc(-c4c(OC)ccnc4)nn3)C2)=O)CCC2(CCNC2=O)CC1 CCCC(C(=O)NCC(C)(CC(C)C)NC(c1sc(C)nc1C)=O)C(C)C Cc1sc2ccccc2c1C(=O)NCC(C)NC(=O)Cc1cnc2ncccn12 CCC(C)CCC(=O)N1CC(C(=O)N(C)CCN2CCOCC2)C(C2CC2)C1 c1(CC)cc(C(=O)N(C2CCCN(C(C3CC3C(=O)OC)=O)CC2)C)c(C)nn1 C(c1cn[nH]c1)=C(C)C(=O)N1CCC1C(=O)N(C1CCCC1)CC(C)C C(=O)(CC(C)(C)C(F)(F)F)NCc1c(N(CC=C)C)cccc1 C1(C(=O)NCCCOCC)C(C2CC2)CCN1C(c1cc(OC)cnc1F)=O N1(C(CCCOCCC)=O)CC(NC(C2OCC3CCCC23)=O)C2(CC2)C1 c1(C(=O)OC)ccc(F)nc1NC(C1CCN1C(=O)CN1C(=O)CSC1=S)=O c1(COC(F)(F)F)c[nH]c2ccccc12.c1(C(C)CCO)ccc(C(F)(F)F)cc1 C1(NC(C(COC)O)=O)CCN(Cc2ccccc2-c2ncc[nH]2)CC1(C)C C1(NC(COC(CC)(C)C)=O)CN(C(c2n[nH]c(C)n2)=O)CCC1(C)C C1(CNC(c2cnc(CCC)s2)=O)CC2(CC(NC(C3CCN3CC)=O)C2)C1 c1(C(=O)NC(CCC(C)C)C)cc2c(s1)CCN(Cc1ccc(Br)c(Cl)c1Cl)C2 C1(O)(CC#C)CC(C(=O)NCC(O)CN(C)C(c2ccnn2C(C)(C)C)=O)C1 C1(C(=O)NCC2CN(C(C(C)(C)F)=O)C2)C2Cc3ccccc3C12 C(=O)(C(C)CC=CC)N(CCOCCNC(C1C(C=C)CC1)=O)C C(C(CNC(=O)Cc1nc([N+](=O)[O-])n[nH]1)C(F)(F)F)NC(c1cncc(C)n1)=O C1(C(CNC(C=C(C)Cl)=O)F)CCN(C(c2cc(C(F)(F)F)on2)=O)CC1 C1(C)(CNC(C(COC)(C)O)=O)CN(C(c2cc(C(C)C)no2)=O)CCO1 C1(CC(=O)NCCN(C(CC(c2c(OC)cccc2)C)=O)C)CC(=O)NC(=O)C1 C(=O)(CCCC(=O)N1CSCC1C(=O)NCC1CCCC1N(C)C)OCC c1(OCC)ccc(C(=O)NC2CCN(C(=O)C=C(CC)CC)C2C)cn1 c1(COC(C(C)(N(C)C(=O)OC(C)(C)C)C2CC2)=O)cc(F)c(O)c(F)c1 S(=O)(=O)(c1ccc(Cl)cn1)NC1CC(C(N2CCOC3(CC3)C2)=O)C1 CC1(C)CC(CNC(=O)CCCn2ccnc2)CN1C(=O)Cc1ccoc1 Cc1nc(C)n(CCC(=O)NC2CC(NC(=O)COCCF)CC2O)n1 C=C(C)C1OCCC1C(N1CCC(n2cccn2)(C(=O)NCC(C)O)CC1)=O CCC(CC(=O)N1CCC(C)CC1C(=O)NCC1CC2(CC2)C1)C(F)F N1(C(c2n(CC)ccc2)=O)CCCC(CCC(=O)NC(C)Cc2ccncc2)C1 C1(C(=O)NCC2(C)CC(NC(=O)C3=CCCSC3)C2)CCc2ccccc2O1 c1(NC(C(C)C)C(C)NC(=O)Cn2cc([N+](=O)[O-])cn2)ncnc2scnc12 c1(OC)cc(C(=O)OC2CCCC2)c(Br)cn1.C12CC1C(=O)NCCNC2=O c1(NCC2CN(C(Cc3cccc(OC)c3)=O)CC2(C)C)nc[nH]c2nccc1-2 C1(OC)CN(C(c2ccc(C)[nH]2)=O)CCC1NCc1ccc(-n2ccnc2)cc1 c1(OCC(=O)NCC2CCCN(C(=O)CCn3cccn3)C2)cccc(Cl)c1 CC1(C)CCC(CNC(c2ccc(CO)o2)=O)N(C(=O)CSS(C)(=O)=O)C1 N1(C(C(C)OCC)=O)CCC(C(N2CC(C(=O)OC)C2)=O)C(O)C1 C12(c3nn(-c4ccc(C)cc4)c(-c4coc(C)n4)n3)CC3CC(CC(C3)C1)C2 C1(C(COC)=O)CC2CCC(C1)N2C(=O)OCCF c1(C(=O)NC(CC2CN(C(C(C)C(C)(F)F)=O)C2)C)cncc2ccccc12 N1(C(C(CCC)N(C)C)=O)C2CCC1CC(NC(C1(C3CCCO3)CCC1)=O)C2 c1(OC)ccc(C#N)c(NC(C2CC2C(=O)Nc2ccccc2F)=O)c1 CC1(CNC(=O)C(F)(F)CN2CCCC2)CN(C(=O)CCN2CCC2)CCO1 c1(SC)cccc(C2CCN(CNc3cccc(C4CC4(F)F)c3)C2)c1 C(=O)(C1CCCn2nccc21)NCCOCCNC(C=Cc1cc(C)c(=N)[nH]c1)=O C1(C(=O)NCCC2CC(NC(C(CCC)C)=O)C2)CSc2ccccc2O1 CC(C)(C)C1=NOC(C(N2CC(CNC(c3ccsc3)=O)C3(CCC3)C2)=O)C1 c1(C(N(CCNC(C2(C(C)(F)F)CC2)=O)CC)=O)cc(CO)oc1C N1(C(C(=O)Nc2c(OC)cccc2)c2ccsn2)CCn2c(nc(C)c2C)C1 CCCC(CCCNC(=O)COc1ccc[n+]([O-])c1)NC(=O)CC1(OC)CC1 C=C(Cl)CC(C(=O)N(C1CC2CCC1O2)C)NC(=O)CCc1ccn(C)c1 C12(C(=O)NC(C)(C)CF)CCN(C(c3c[nH]cc3C3CC3)=O)CCC1C2 c1(CC(C(=O)NC2C(C(=O)OC)CCCC2)N)ccc(OC)c(F)c1 C1(CCCCNC(CCOC)=O)CCN(C(=O)C(C2CCCOC2)OC)CC1 CN1CCC2(CCN2C(C2C3CC4C(C3NC(=O)CC3COC(=O)C3)C24)=O)C1 C1(CNC(c2c(C)snn2)=O)CC2(CCN(C(c3cccc(CO)c3)=O)CC2)C1 C1(C(=O)NC2CC(CCNC(c3cccc(CCC)c3)=O)C2)CC(=O)C12CCC2 CC1CN(C(=O)COC2CC(NC(C3CCCC4(CC4)C3)=O)C2)C(C)C1C c1(C(=O)NC2CN(C(c3ccc(CO)o3)=O)CCC2F)cc2ccc(O)cc2[nH]1 C(=O)(C=C1SCC(=O)N1C)N1CCN(C(C(COC)C)=O)CC1C1CCC1 C(=O)(C1Cc2ccc(F)cc21)NCCCN(C)C(C1CCCN1C1CCCC1)=O c1(N(C(=O)CC2CCCN2C(=O)COCC(F)(F)F)CCC#N)cc(Cl)ccc1Cl c1(C(CC)N(c2cc(C)ccn2)C(=O)CSc2ccco2)cccc(C)c1 CCCCCCCCOCC(N1CC2(CC2)CC1CNC(=O)C(C)S(N)(=O)=O)=O c1(C(=O)NC2CCC(CNC(c3cc[nH]n3)=O)C2)cc(Cl)c(F)cc1F C1(O)(C(C(=O)NC(C)CC2CCCCC2)NC(CC2C(CC)C2)=O)CCCCC1 c1(C(C)OC)cc(OC(CO)C(=O)N2CC(Cn3cc(CN)nn3)C2)ccc1Cl c1(C(N2CC(C(=O)Nc3cn(CC)nn3)C(O)CC2)=O)cncc2ccccc12 CC1CC(C(=O)NCC(C)(F)CNC(c2cc(C3CC3)no2)=O)CC(=O)N1 c1(C(N2C(C)(CC)CC(NC(=O)CCCOC(C)=O)C2)=O)ccc2c(c1)OCC2 C1(O)(C(C)NC(CC=CC=C)=O)CCN(C(=O)CCC(C)C)CC1 C#CCC(C)(CNC(=O)COC1CCN(C(c2cnco2)=O)C1)CO CC1CN(C(C2CCCN2C)=O)CCCN1C(=O)CCCNC(N)=O c1(OC)c(C(=O)N(C(C)CCNC(c2cncc(C(N)=O)c2)=O)C)ccnc1Cl Cc1cnc2c(C=O)cccn12.N1(C(C2CC23CC3)=O)CCN(C)CC1CCO c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(=O)CC3(CO)CC3)CC1CO)CC2 CN1C(=O)NC(=O)C12CCN(CC1CCCC3(CCC3)C1)CC2 S(=O)(=O)(c1ccc(NC(F)F)c2cnccc12)NC1C(C(N)=O)CCC1 C(C)(C1OCCc2sccc21)N(C(C(=O)NC(c1c(C)nc(C(C)C)s1)C)=O)C CCN(OC)C(=O)CNC(=O)C(Cn1cccn1)NC(C1CC(C)(C)CO1)=O c1(C(=O)NC2CCCCC2CNC(c2n[nH]c(O)n2)=O)ccc2nc(Cl)nn2c1 C#Cc1ccc(C(N2CC3CC2C3C(=O)Nc2nc(Cl)cnc2Br)=O)c(Cl)c1 Cc1ccc2c(c1)CN(C(C1C3CN(C(=O)COCC(F)(F)F)CC13)=O)CC2 C1(N(C)C)CCC(C(=O)NCC2CCC(NC(c3ccc(F)cc3)=O)C2)CC1 C1(C(=O)NCc2cc(COC)no2)CN(C(=O)Cc2cnns2)CCC1(C)C N1(C(Cc2[nH]cc(C)c2)=O)CCC(CNC(c2ccncn2)=O)C(F)(F)C1 Cc1nc2n(n1)CC(C(=O)N(CCNC(c1coc(C#N)c1)=O)C(C)C)CC2 c1(C(=O)OCC(=O)N(CCC)C2CC2)cn2cc(Cl)ccc2n1 C1(NC(C2CCCCC23CCC3)=O)CCN(C(=O)CC2CCSC2)CCC1CO c1(C(=O)OCCl)ccccc1OC1CC1.CC(C)(C(C)NC(c1ccncc1)=O)O N1(C(CCc2ccc(C)o2)=O)CCN(C(c2csc(-c3cnc[nH]3)n2)=O)C(C)C1 C1(C(N2CC(CCC)C2)=O)CCC(C)(C)N(C(C2CC2Cl)=O)C1 CCC(C)CC(C(=O)NCC(C(C)C)C(C)C)NC(C1CCCC(=O)C1)=O c1(C(=O)NCC(C2CC2)NC(CC2CCC(C)O2)=O)cccc(C2(C#N)CC2)c1 C1(NC(=O)CC2CCOC2)CN(C(c2cocn2)=O)C2(CCCCC2)C1 C(CCCCNC(=O)C(C)Cc1ccccc1)NC(C1(C#C)CC1)=O c1(C(=O)NCC(CC)NC(C2CCCCNC2=O)=O)c(F)ccc(C)c1F c1(N(C(=O)CC23CC(C2)C3)CCN2CCC(CC)CC2)cc(C)ccc1[N+](=O)[O-] C1(C(=O)NCCCC(CO)NC(CC(C)(C)O)=O)CCC(=C(F)F)CC1 C(=O)(C1CCc2nccn21)NC(C1CCN(C(c2c(CC)noc2)=O)C1)C c1(CC)ccc(C(=O)NCCN(CCOC)C(c2cscc2CC)=O)c(OC)c1 C(=O)(C1=CC2CC=CCC12)N(C1CCCCCC1)CC C1(NC(C2CCN(C(c3ccc4ccoc4c3)=O)C2)=O)CCC2(CCC2)CC1 C1(C(=O)NCC(C(C)C)(C)O)CC(F)CCN1C(c1cc(O)cc(=O)o1)=O c1(C(=O)NC(C)CNC(=O)CCC(O)C(C)(C)C)cc2c(nn1)OCCS2 S(=O)(=O)(c1ccc(C#N)cc1)N(C(CC#C)CC)CCC.C1C(=O)N1 Cc1nn(CC(=O)NC2COCCN(C(=O)Cc3nc(C)c(C)o3)C2)c(C)c1Cl n1(C(C)C)ncc2cc(C(=O)NCC(C)(C)NC(=O)C(F)C3CCOC3)cnc12 C(=O)(CC(C)CC(C)C)N(CCC)CCNC(=O)CCc1nc(C(F)(F)F)n[nH]1 c1(C(N(C)CC2CN(C(c3c(C)nco3)=O)CC23CC3)=O)cccc2nc[nH]c12 C1(CC(C)CNC(C2CCC(C3CCNCC3)O2)=O)C=NN(C)C1=O Cc1ccc(C(=O)N2CCC(C(=O)NCCc3cccc(O)n3)O2)cc1C#N C1(C(=O)NC(C)CCNC(=O)CCCc2cnccn2)CCCCN1S(C)(=O)=O N1(C(CCCN(C)C)=O)CCC2(CCCN2C(=O)CC2CC(O)C2(C)C)CC1 c1(NC(=O)Nc2cccc(SCCC)c2)cc(S(N)(=O)=O)ccc1Cl N1(C(=O)NCC(=O)OCC)CCC2(CCCC2N2CCCC(C)(C)C2)CC1 c1(NC(C2C(CCC)CNC2)=O)ccnc(C)c1C.C(C)(C)(C(=O)OC)SCC C1(CC)(CNN2OC(C)(C)CC2)CCN(C(=O)OCC)C1.c12cccc(c1)O2 c1(C(N2CCC(C3CCCN3C(=O)C=CBr)C2)=O)cc2c(s1)CCC2=O N1(C(CN(C(COC)=O)C)=O)CCCC2(C1)CC=CCCCN2C(=O)CNC=O N1(C(CC(=O)NC2CC2)=O)CCC2(CO)CN(C(=O)CC3CCC3)CC2C1 C(=O)(CCCCCC(C)(C)C)NCC1CN(C(c2c(COC)noc2)=O)CC1C c1(C(C)OC(c2cn(-c3cccc(Cl)c3)cn2)=O)ncccc1Br N1(C(c2ncn(C(C)C)n2)=O)CC(CNC(=O)Cc2cnoc2)OC2(CCC2)C1 C1(NC(COCCC)=O)CC2CC1N(C(C1CCCC(C)(C)C1)=O)C2 c1(C(=O)NC(C)C)c[nH]c2ccccc12.C1(=O)C(C(C2CCOC2)C#C)CN1 C1(CCNC(c2cc(C)n(C)c2)=O)CC(F)(F)CN1C(=O)C(C)C1CCC1 Cc1nn(CC(=O)N(C2CCC(NC(=O)CS(C)(=O)=O)C2)C)cc1[N+](=O)[O-] c1(NCCCC(C)NC(c2ccoc2Br)=O)snc(Cl)c1C#N C1(CC(=O)CCN(C(=O)CCS)C)CCC(=O)NC1.C(CCNC(C1CCC1)=O)O C(N=c1cc[nH]c(C(=O)O)n1)C1CCN(C(=O)CCCCC2CC2)C1 N1(C(C(C)SCC)=O)CCOC2CN(C(c3csc(C(=O)OCC)n3)=O)CC12 N1(C(c2ccc(C)o2)=O)CCN(C(=O)C2=C(Cl)CCOC2)C(C)CC1C c1(N2CCC(NC(C(CCCC)O)=O)C2(C)C)ncnc2c(Br)nn(C)c12 C#Cc1ccc(C(=O)NC(C)C(C)CC(=O)NC(C)(CC(C)C)C(N)=O)c(C)c1 C1(CC)(NC(=O)CC2CC(CF)C2)CCN(C(C2CC2(F)Cl)=O)CC1 C1(CC(N2CC(C)(CSC)C2)=O)CC(O)CN1C(=O)C(C)O C(=O)(C1=NOC2(CCC2)C1)NCC(C)(C)CO.C12CCN(C13CC3)C2=O CCCC(C(=O)OC)NC(=O)NCCOc1cc(C(F)(F)F)nn1C(C)(C)C C1(C(=O)NC(C(C)NC(=O)Cc2csc(-c3ccco3)n2)C)OCCOC1(C)C c1(C(N2CCCN(c3ccnc(C)n3)CC2)=O)cc2cc(Br)ccc2[nH]1 c1(OC)cc(F)c(S(=O)(=O)N2CCOCC2CC(F)F)cc1Br N1(C(c2n(CC)nc(C)c2)=O)CCC2(C=C(C(=O)NCCSCCO)C2)C1 C1(CNC(c2ccn(C3CC3)n2)=O)COCCN1C(c1cncs1)=O Cc1cc(C(=O)NCC2CCCN2C(=O)COCc2ccnn2C)ccc1F C1(CNC(C(C)OCCOC)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 Cc1nc(C(=O)NC2CCN(C(=O)CCC3(C)CC3)C2C(C)C)cn1C N1(C(C2C(C)N(C(c3ncccc3F)=O)CCC2)=O)CCc2n[nH]cc2C1 N1(Cc2cc(C)c(C(F)F)cn2)CC2(COC(=O)N2C)C1 c1(OC)cc(C(N2CC(COC)CC2CNC(=O)C(C)(C)C2CCC2)=O)ncn1 C(C)(C)(CCCNC(c1ccc(-c2cccs2)cn1)=O)NC(CN(C)CC)=O Cc1cc(C(N2CC=CC(NC(=O)C(c3ccncc3C)C)C2)=O)c(C)cn1 c1(C(C)C)cccnc1CC(=O)N(CCCNC(=O)COCC1CC1)CCO c1(C(=O)OC)no[nH]c1=NC(=O)C1CCN(Cc2csc(C)c2C)CC1O C=C1CC(C(=O)NC(C(O)CO)C2CC2)(CNC(C2CC=CCC2)=O)C1 N1(C(CC2ON=C(C)C2)=O)CCC(NC(c2cc(Br)sn2)=O)C(C)(C)C1 C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(C2CC(O)C2)=O)C2CCN1C2 CCCCC(CNC(=O)C=Cc1cnc[nH]1)NC(c1cc(Cl)c(Br)[nH]1)=O Cc1c(C(=O)N(CC(C)C(=O)NC(CO)C(F)(F)F)C)cccc1O Cc1cc(C(N2CC(NC(c3c(C)noc3C(F)(F)F)=O)C(C)C2)=O)cc(Cl)n1 c1(C(N2CC(C(C)NC(C3CC3C(C)(F)F)=O)C2)=O)n[nH]cc1C1CC1 C1(C(N2CC=C(C)CC2)=O)CCN(C(c2c[nH][nH]c2=N)=O)CC1(C)C C12(C(=O)NCC3N(C(CCc4nnc(C)o4)=O)CCC3)CCC(O)(CC1)CC2 CC(CS(C)=O)C(=O)NCCCNC(c1cnc(O)c(Cl)c1)=O C1(C(=O)NC23CC(C(=O)NCC(=O)OCC)(C2)C3)CC2C=CC1O2.C(C(=O)NC)OC N1(C(C2C(C(C)=O)C2(C)C)=O)CCN(C(C2CCCC3CC23)=O)CC1C c1(OC)cccc(C)c1-c1ccc(C(=O)NCCOC2CCCC2)nc1 C(=O)(C(F)(F)CCn1ccnn1)N(C)CC1(CNC(C2(C)CC=CCO2)=O)CC1 C1(C(N2CCCC2CNC(=O)CC2CCC(=O)C2C)=O)(CC)CC(F)(F)C1 N1(C(CCCSC)=O)CC2(C1)C(NC(C1CCS(=O)(=O)C(C)C1)=O)CCS2(=O)=O N1(C(=O)NCC23C(CN(C(=O)OC(C)(C)C)C2)C3)CCC2COCC2C1 C1(NC(CCCC)=O)CC(NC(=O)CC(c2c(C)noc2C)C)C(O)C1 CN1CCCCC1C(=O)NCc1nc(CC(=O)NCC2(F)CCN(C)C2)cs1 N1(C(CC=CCC)=O)CCCC(O)(CCNC(c2cc(C(F)(F)F)ccn2)=O)C1 O=C(CCN=c1[nH]ccs1)NC1(CSC)CN(C(=O)CCN2CCCC2)C1 C1(O)(CCNC(=O)CSc2ccccc2)CCN(C(C2(OCCO)CC2)=O)C1 C1(NC(C(COC)C)=O)CCC(NC(=O)Cc2ccc(C(=O)OC)nc2)CC1 N1(C(C2(C3CC3)CN(C(C3(OCC)CC3)=O)C2)=O)CCC2OCCC2C1 N1(C(CCC(N)=O)=O)CCC(C2CC(NC(=O)Cc3ccc4sccc4c3)C2)C1 N1(CC(N2C(C)(CNC(Cc3n[nH]c(=NC)s3)=O)CCC2)=O)C(=O)CNC1=O C12(C(=O)NC(C)CCNC(=O)CCCCc3ccccc3O)CCC(F)(CC1)C2 N1(C(COC(C)C)=O)CCC(O)C(NC(=O)C=C2CCC(C)CC2)C1 C(C(=O)NC1NC(=S)N(c2cccc(C)c2)C1=O)(C(C(C)C)OC)OC C1(CCC)CN(C(c2cncc(F)c2)=O)CCN1C(c1ccnc(CO)c1)=O C1(CC)C(C(=O)NCc2cccc(OC)n2)CCCN1C(=O)C(O)CCN(C)C N1(C(CCCn2cc(CCC#N)nn2)=O)CCC(F)(OCCO)CC1 CN1CC(O)CC1C(=O)NC1CC(NC(=O)Cc2ncc(Cl)s2)C1 C1(SCC)CCCC1N=c1nc2sccc2c(NCc2nc(Br)cs2)[nH]1 C1(CN(C)C(C2CCC(=O)O2)=O)CCN(C(c2ccnn2CC2CCC2)=O)CC1 c1(C(=O)NCCC2(NC(CC3ON=C(CC)C3)=O)CC2)ncc2c(F)cccn12 C(c1cccnc1)=CCCCn1cc(C(C)(C)N(C(=O)CCS(C)(=O)=O)CCO)nn1 C1(CNC(c2c(C)cccc2)=O)COCCN(c2cc(O)nc(C)n2)C1 Cc1cc(=NC(=O)c2cnc(-c3ccc(O)cc3F)cn2)[nH][nH]1 c1(C(C)C)nn(C)cc1C(=O)NC1COCC1NC(C1(c2cc[nH]n2)CC1)=O c1(NC2(C(=O)NC3CC(C(F)C(=O)N(C4CC4)SC)C3)CC2)ccccc1Br N1(C(C(C)OCCC#C)=O)CCC(C2CC2)(NC(=O)COc2cccc(F)c2)C1 CCCCCC(O)C(=O)NC(C1(CNC(c2cn(C)c(=O)c(C)n2)=O)CC1)C c1(OC)ccc(C(=O)NC(C2CN(C(=O)C=Cc3cn(C)cn3)CCO2)C)nc1 N1(Cc2ccc(C(=O)O)s2)CCC2C(CCN2C(c2cc(O)c(O)c(O)c2)=O)C1 C(=O)(C1CCC(=O)c2ccccc21)C(=O)CCCC(N)=O.C(C(C)(C)N)NC N12CCCC(COC)(C1)C2=O.C1(CCC)(NC(C2CC2COC)=O)CCNC1=O c1(NC(C2CCN(C(C(C)=O)=O)C2)=O)ccnc2c(Br)cccc12 C=CCC(CC(C)C)C(=O)N1CC2CCC(C1)N2C C(=O)(C(C)Cc1ccco1)NC(CC)CNC(=O)CNC(=O)NC1CC1 c1(-c2cc(CNC(c3n(C)nc(-c4ccccc4)c3)=O)[nH]n2)ccc(F)cc1O c1(C(=O)OC)oc(C(=O)NCC(F)CNC(C2(C)CCCO2)=O)cc1C C12(NC(c3ccsc3C(F)(F)F)=O)CCCC1(F)CN(C(C1CCCOC1)=O)C2 Cc1ncccc1CCC(=O)NCCC(C)(C)CNC(c1ccc(Cl)cn1)=O C(=O)(C(C(C)C)C(C)C)N1CCC(OCCNC(C=Cc2c(C)cccc2)=O)C1 c1(CC)ccc(OCCC(N2CC3CC2C3NC(=O)CCCCSC)=O)cc1 CC(C)CC(C(=O)N1CCCOC(CNC(C2CSC2)=O)C1)C(N)=O c1(C(=O)NC(CC2CN(C(C=CC)=O)C2)C)cc(F)c(CO)c(F)c1 c1(C(=O)NCC2CCC(NC(=O)C#CC3CC3)CC2)c(Cl)ccc2ccncc12 C1(C(N2CC3(CN(C(C(CCC)C)=O)C3)C2)=O)CC12CCC(=O)CC2 Cc1ccc(NCC23CC(C#N)C(C2)C3)c(F)c1F CC1CC(NC(=O)CNC(=O)C2CC2)CN(C(c2occ3c2CCC3)=O)C1 C1(C(=O)NCC(C)NC(c2nccn3nccc23)=O)C2Cc3ccccc3C12 CON(CCC(=O)NC(C)(CCO)C(F)(F)F)C(=O)C(C)n1ccnc1 c1(CNC(=O)NC(CCC=C)C2CC2)cccc2c(O)ncnc12 N1(C(c2nc(C)oc2)=O)CCCN(C(C23CC(CCO2)C3)=O)C(C)C1 c1(CC(CC)NC(=O)C(c2cccc(C(F)(F)F)c2)N)ccc(Cl)cn1 N1(C(c2c(C)ccnc2C)=O)CCC2C(CCCN2C(c2cn(C)c(O)n2)=O)C1 N1(C(c2c(C)ccc(F)c2)=O)CCc2cc(C(=O)NCCC(N)=O)ccc2C1 N1(C(C2CC=CC2)=O)CCC(C2CCCN(C(C3CC=CC3)=O)CCC2)CC1 C1(NCCC(CNC(CC)=O)O)CC(C(F)(F)F)CN(C(=O)OC(C)(C)C)C1 CC1CCC(CC(=O)NC2CC(NC(c3ccccc3OCCBr)=O)C2)CC1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CC2C(CNC(=O)CC3CC34CC4)C2C1 C1(CNC(CN(C)C)=O)(NC(=O)CCc2nnc(C3CC3)o2)CCOC1 CC1CC(=O)NCC1C(=O)NCCCOCCN(C(=O)CCCCCO)C C(=O)(C1(C)CC(=O)N(C)c2ccccc21)NC(C(C)C)CCNC(=O)CC1CC1 c1(C(N(CC(C)NC(C2(C)CCC(=O)C2)=O)C)=O)cccc(=O)n1O N1(C(C(C(C)(C)C)O)=O)CC(NC(=O)C=C(C2CC2)C2CC2)CC12CCC2 C1(C(=O)NC(C)CNC(=O)CCCc2cccs2)CC(C(=O)OC(C)(C)C)=NO1 C=CC1CN(C(c2ccnc(C)c2O)=O)CC1NC(=O)C(C)OCC(C)C c1(OCCCC)ccc(NC(=O)NCC2(C)CCCN(C(=O)CSC)C2)c(Cl)c1 N=c1[nH]c(N2CC3(CN(C(=O)OC(C)(C)C)C3)C2)nc(N)c1[N+](=O)[O-] n1(CC)ccc(C(=O)NC2CN(C(=O)CC3CC4(CC4)CO3)CC2(C)C)cc1=O c1(OCC)ccccc1NC(C1C=CCCN1C(=O)C(O)CN1CCCC1)=O N1(C(CN(C(=O)CSCC(F)F)CC#C)=O)CC2(COC(=O)N2C)C1 N1(C2CC3CN(C(=O)OC(=O)C=Cc4cccs4)C2C3)CCc2cccc(Cl)c2C1 N1(C(CCC)=O)CCC(CCC(=O)N(C)CC2(O)CCOC2)C1 C(=O)(N=c1ncc(Br)c[nH]1)NC(C)Cc1ccn(C2(C(F)(F)F)CC2)n1 CC(C)C(C(=O)NCc1ccn(CC(F)F)n1)N(C)C Cc1nc(NC2CCN(Cc3cc(N(C)C)ccn3)C(C)C2)c2ccsc2n1 Cn1cc(CC(=O)NCC2(C)CC(NC(C3CCO3)=O)C2)cn1 c1(NC(=O)C(CC)OC)cccc(N(C(=O)C#CCN(C)C)CC=C)c1 C1(NC(c2c(CC)nc(C)nc2)=O)CCC2CCN(C(C3CCCC3O)=O)C1C2 C=CCC(C)(C)C(=O)N1CC2(C(=O)NCCc3ccccn3)CC1CO2 c1(C(N2CCC(C(=O)NCC(CC)F)C2)=O)ccccc1NC CC(=O)CCCCC(=O)N1CCCC1C=CC(=O)N(C)CCC1CC1 C1(CC(=O)NCC(=CC(=O)N(CC(C)(C)O)CCC)C)CCCCC1 C(C)(C)(CC(C)N=c1ccnc(NC2C(C3CC3)C2(F)F)[nH]1)OC N#Cc1c[nH]c2ncnc(NCC3CC(C(=O)Nc4ccc(Cl)c(CO)c4)C3)c12 C1(CNC(c2csc3nnsc23)=O)(NC(C2CC2C(F)F)=O)CCC(F)(F)CC1 c1(OC)cc(C(N2CCCCC(NC(C3(CF)CC3(F)F)=O)C2)=O)cc(F)c1 c1(C(N(CC=CC(=O)N(CC)CC2(O)CCC2)C)=O)cc(C)ccc1O c1(C(=O)NC2CCCN(C(C(CC)O)=O)CC2)cc2cc(C)ccc2s1 c1(C(N(C2CC2NC(C2(Nc3ccccc3)CC2)=O)C)=O)cc(C2CC2)on1 C(=O)(CCCCN=c1nc(N2CCC3(CC(F)C3)C2)c2c([nH]1)c(C)nn2C)NC CC(CNC(=O)CN(C(=O)CCC1(C)CC1)CC1CC1)CC1CCC1 N1(C(C2CN(C)C(=O)N2)=O)CCCC2(CCN(C(C3CC(=O)C3)=O)C2)C1 Cc1ccc2occ(CC(=O)NC3CC3CNC(=O)Cc3sc(O)nc3O)c2c1 C#CCCC(O)C(=O)NCC1(C(N)=O)CN(C(=O)CCCN=[N+]=[N-])C1 c1(C(=O)NC(CCCNC(c2ccn(CC(C)C)n2)=O)C)csc(S(N)(=O)=O)c1 Cc1c(O)ccc(C(N2CC3C(NC(=O)Cc4csc5cncn45)C3C2)=O)c1C c1(C(=O)NC2CCCC(C(=O)NC(CC=C)CC)C2)nnc(O)nc1O N1(C(CC(C)CF)=O)CC2(CCN(C(c3ccnn3CCN(C)C)=O)CC2)C1 C1(=O)C(CCC)C(=O)C(=O)CCN1CC#C.C1(N)CCC(C2CC2)C1.OCC C(CC(C)C(=O)N1CC2CC2(CNC(=O)CNC(C)=O)C1)OC N1(C(C(C)=C(C)C)=O)CCC(C2(O)CCN(C(=O)C(C)(Cl)Cl)C2)CC1 C(=O)(C(CC1CCCCC1)NCc1cn(C2CCC2)nn1)OC C12(C(N3CC4=C(CN(C(C5CNC(=O)N5)=O)C4)C3)=O)CCCCC(=O)N1CCC2 C12(C(N3CC(C#N)C3)=O)CC(CN(C(=O)CCCn3cncn3)C1)C2 CCC(CC)(CN=c1[nH]c(C2CC2)nc(C)c1Br)NC(c1cccc(Cl)n1)=O N1(c2nccc(C)n2)CCOC2(CCN(C(=O)CCC3CC3(C)C)CC2)C1 C(C)(CCS(=O)(=O)NC1(CO)CCCC2CC12)OC CC1(C(=O)NC2CC(CCF)C2)CCN(C(=O)CN2CCNC2=O)C1 N1(C(c2ccc(C)[nH]2)=O)CCC(C(=O)N(C)C(c2ccccc2F)C)C(C)C1.CO c1(C(N(C2CCC(CC)CC2)C(=O)C(C)SC2CC2)=O)cn2ccsc2n1 C1(O)(CN(C)C)CCCN(C(=O)NCC2CCC(F)CC2)C1 CC1CCN(C(c2ncncc2Cl)=O)CCN1C(=O)CCOCc1ccccc1 N1(c2ncc(OC)cn2)CCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)CC1C C(C(=O)NCC1CCCC(NC(=O)Cc2nc(CC)cs2)C1)(C(C)C)OCC Cc1c(-c2cncnc2C(=O)Nc2cccc3ncsc23)ccc(Br)c1F C1(C(C)C(=O)N(C)CCOCCN(C(=O)COC2CC2)C)CCCOCC1 C#CC1(C(N2CC(CN(C(=O)C(C)(C)OC)C)C2)=O)CCCC1 Cc1cncc(C)c1C(=O)NCC1CCN(C(=O)CCCc2cccnc2)CC1 c1(C(=O)Oc2ccc(C(=O)NNC(=O)C3CCCCC3)cc2)ccc2cncn2c1 C1(C(C)NC(c2cccnn2)=O)CCCC(NC(c2cc(C3CC3)nn2C)=O)C1 c1(CC(=O)N(CCC(C)NC(=O)C2=NOCC2)C)cccc(C(F)(F)F)n1 c1(OC)cc(F)cc(C(=O)NCCNC(c2sc(F)cc2Br)=O)c1N C(=O)(CS(=O)(=O)NC(=O)C(C)SC1CC1)NC1C(COCC)CCC1 C1(C(=O)NCCC2CN(C(CS(CC)(=O)=O)=O)C2)CCCN(S(N)(=O)=O)C1 CC(C)(C)CC(=O)NNC(=O)NC1CCCCC1(C)C c1(C(c2n(C(C)C)nnn2)NC2CC(Cl)(Cl)C2)cc(F)ccc1Br c1(C(N2CCC(O)(C(=O)N(C)C)C2)C)ccc(Br)cc1F Nc1cc(C(N2CC=C(CNC(=O)CC(F)(F)F)CC2)=O)ncc1F CC1CN(C)C(=O)CN1N1CCC2(CC1)CN(C(c1cn(C)nn1)=O)CCO2 CC(C)CCC(C(=O)NC1CN2CCCC1C2)NC(=O)CSC(F)(F)F c1(Cc2cn(C(CC)C(=O)N3CCC4CC34)nn2)cc(F)cc(F)c1 c1(OC)cc(OC)nc(N2CCCC(CO)C2)n1.C12CN(CCS1)C2 C=CC1(CC(=O)N(CCC)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC)CCCCC1 c1(OC)cnn(C)c1C(c1nnnn1C1(C)CC1)NC(C)Cc1ccc(O)cc1 C1(CN(C(=O)CC2(CO)CC2)C)CN(C(=O)C(O)CCn2cncn2)CC12CC2 c1(OC)cc(C(=O)NCC2CCC2NC(=O)Cc2c[nH]nc2C)sc1S(N)(=O)=O c1(C(=O)NC(CNC(C=Cc2cn(C)nn2)=O)(C)C)cc2ccncc2[nH]1 c1(OC)ccccc1CC(=O)NCC(O)CNC(c1onc(C)c1C)=O c1(C(=O)NC(CCCCNC(COCCCOC)=O)C)ccnc(Cl)c1Cl C1(CC)CC(C(N2CC(C)(CCC(N3CC4C=CC4C3)=O)C2)=O)CCO1 N1(C(C#CCNC(CC(CC)C)=O)=O)CCOC(C)CC1 N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)(CNC(c2nnc(C)s2)=O)C1 N1(C(C2CCCCS2)=O)CCC(NC(c2cccnc2)=O)C(O)C1 Cc1ccc(C(N2CCC3CC23C(=O)NCCC(C)C(F)F)=O)nn1 C(=O)(CCC(F)(F)F)N(CCN(C(C1(OC)CC(CF)C1)=O)C(C)C)C C1(COC)(CNC(C2CCC(C)O2)=O)CCN(c2ccnc(SC)n2)CC1 C1(C(=O)NCC2CC(C)(C)CO2)(CC)CCCN1C(=O)CC1(O)CCOCC1 c1(CC(CNC(=O)NC(C(=O)O)c2cccs2)O)ccccc1Br C1(C(=O)Nc2cnc(OCC)s2)C=CCN(C(C23COC(CO)(C2)C3)=O)C1 C(F)(C(=O)N1CCCCCO1)=C(C)CSC1(C(=O)N(C(CO)CO)C)CCC1 CS(=O)C1(CNC(=O)COC2CCN(C(c3cscc3Cl)=O)C2)CC1 c1(C(=O)NC(C)CCCNC(C2(C)CC(C)(C)C2)=O)ncn2c1CCC2 CON1CCC(C(=O)NCCC2CCCN(C(=O)Cn3cccc3)CC2)CC1 n1(CC(=O)NCC(C)NC(=O)CN2CCC(C(N)=O)C2)ncn2nccc2c1=O N1(CCN2CCC(C)(C(=O)OC)C2)Cc2ccccc2OC1=O CCC(CC)C(C)C(=O)N1CC(CNC(=O)C(c2cccc(C)c2)O)C1 C(CCCCC(=O)N1CCCC1C)N(C(c1cc(CC)[nH]n1)=O)C CC1CN(C(c2cc(Cl)c(Br)cn2)C(=O)NCCC2CC2)Cc2c[nH]nc21 C(c1cncnc1O)=CC(=O)NC(CNC(c1c(C)scn1)=O)(C)CO Cc1nccn1CCC(=O)NCC1CCC(NC(=O)C(C)CO)C1 N1(C(C(N2CCC(OC)C2(C)C)=O)=O)CC2(CCC(O)CC2)C1 C1(C)(NC(C)=O)CCN(C(=O)C(C)N(C2CCC2)C(C23CCC(C2)OC3)=O)C1 C(=O)(C(C(C)NC(c1ccc(CC#N)cc1)=O)C(C)C)N1CCC(SC)C1 c1(C(=O)OCC)cc(C(=O)NC2CCC(NC(C)=O)C2)ccc1C C1(CC(=O)NCCC2(CNC(C(C)NC(=O)OC)=O)CCC2)COCCO1 C(=O)(C1=C(Cl)CCCC1)N(CC(=O)NC1CC(=O)N(C2CC2)CC1)CC#C C1(C(C(=O)NCC2C=CC(NC(c3cc(C)on3)=O)C2)O)CCCCCC1 Cc1c(C(N2CCC(CCCNC(C3C4CCC34)=O)CC2)=O)ccn1C c1(C(C)C(=O)NCC2(O)CC(NC(=O)Cn3cccc3)C2)ccc(F)c(F)c1 c1(CNC(C2CCC(OC)CC2)=O)ccc(F)c(Cl)c1N.C12CCN(C1)C2=O C1(C(NOCCCCCNC(=O)C(C)N2CCCC2)=O)(CC#C)CC2(CC2)C1 c1(C(=O)NCC(C)CNC(c2ccccc2OCC#N)=O)c(F)ccc(Cl)c1N N1(C(Cc2n(CC)ccc2)=O)CCC(NC(=O)COC2(C)CCC2)C1C(C)C C(=O)(N1OC2CCC1CC2)c1c(CNC(=O)Cc2ccnc(O)c2)cccn1 c1(C(=O)NC2CN(C(c3[nH]n(C)c(=O)n3)=O)CC2(C)C)cc(F)c(F)cc1Cl C(=O)(C#CC1(C)COC1)NC1CCC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1 N1(C(C=CCCC)=O)Cc2ccccc2C(NC(=O)Cn2nnc(=O)[nH]2)C1 CC(CC(=O)NC(CNC(c1ccc(-c2cc[nH]c(=N)c2)o1)=O)C1CC1)C(F)F c1(CC)cc(C(=O)NC(C2CCOC2)CNC(c2cnns2)=O)ns1 C1(C(=O)NC2(C)CN(C(c3cc[nH]c3C3CCC3)=O)C2)CCCC(F)(F)C1 C1(NC(c2cccnc2C2CC2)=O)CN(C(=O)C=Cc2ccsc2)C2CC12 C(=O)(C1CCc2ccc(Cl)nc21)NCC1(NC(c2nc(NC(C)=O)sc2)=O)CC1 c1(C(N2CCC(C)(C#N)C2)C(=O)NCCC#N)ccc(F)c(F)c1Br N1(Cc2ccc(OC)c(CO)c2)CC2(CCCC2NCc2nnc(C(F)F)o2)C1 C1(C(N2CCC(SC)C2)=O)CN(C(C2OCCCO2)=O)CC1(C)C CC1CCC(CC(N2CC(C(C)NC(C34CCCN(CC3)C4)=O)C2)=O)CC1C N1(C(C2C(C(=O)OCC)C2)=O)CC2CC(C1)N(C(c1cnc(CC(C)C)s1)=O)C2 Cc1cccc(C(O)C(=O)NCC2CN(C(C3NC(=O)C4CC34)=O)C2)c1F C1(C(=O)N(C2CC2)Cc2cccc(C)n2)(NC(C(C=CC)O)=O)CCC(C)(C)C1 C(N=c1nc(NC2CCN(S(C)(=O)=O)C2)c2c([nH]1)c(C)nn2C)c1n(CC)ncc1 N1(C(C2(C(C)C)CC2)=O)CC(NC(c2cnoc2-c2ccc(F)cc2)=O)C(C)C1 c1(OCC)cc2c(cc1NC(=O)C(=O)NCCC1CCCO1)OC(C)C2 c1(C(N2CCC(NC(C3CCCN(CC)C3)=O)C2C)=O)cc(C)c(C#N)cn1 CCCC(C(=O)NC(C)CN(C)C(C1(NC(C)=O)CCC1)=O)NC(N)=O c1(OC(C)C)ccc(S(=O)(=O)N2CCC(C(C)C)CC2)cn1.C1C(C)C(=O)N1 C1(NC(=O)OC)CCN(C(=O)C(C)N(C)C(C2CC23CC3(F)F)=O)CC1 N1(C(C=CCCC)=O)CCC(C2CCN(C(c3ccnc4[nH]nnc34)=O)C2)C1 c1(OC)ccccc1OC(C)C(=O)N(CC(C)O)CCNC(C1C2(CC2)C12CC2)=O CC1CCCCC1C(C(=O)NCC1(C)CCCCC1)N1CCC1c1cccc(Br)c1 Cc1cccc(CC(=O)NCCC2CC(NC(C3CCNC3=O)=O)C2)c1 c1(C(=O)NCC(CC)NC(=O)C(C)(C)C2(C)CC2(F)F)cccc(Cl)c1N Cc1ccc(C(=O)N(C2CN(C(c3cnnc(O)c3)=O)CC2(C)C)C)cc1Cl C1(CO)CCCCN(Cc2cn(CC3CC(c4ccccc4)CO3)nn2)C1 C(C(C)C(F)C(=O)NCCSC(C)C)NC(C(C(C)C)SCC)=O Cn1cc(C2CCN(C(C(=O)N(C(C)(C)C)CC3CCCO3)c3cnsc3)C2)cn1 N1(C(CCOCCCOC)=O)CCOC(CCNC(=O)C(O)C2CCC2)C1 CC1(C)C(CC(N2CCC(CO)C2)=O)CCN1C(=O)C(O)Cn1cncn1 C1(CNC(c2cccc(SCC)c2)=O)CCN(C(=O)C2=COCC2)CC1(F)F C=CCCC(C)NC(c1sccc1CNC(C1CCCN1C(C)=O)=O)=O C(CC(C(C)C)NC(=O)Cc1nc(C2CC2)cs1)N(C(c1cc(CC)no1)=O)C N1(C(=O)NC(=O)OC)CC(C)N(C(C23CCC(CC2)C3)=O)C(C)C1.C1CO1.C(COC)N CCCCC(C(=O)NC)NC(C1CN(C(C2(OC)CCCC2)=O)CC12CC2)=O N1(C(C2CCCCN(C(C(CC)CC)=O)C2)=O)CCC(C)(C2CC2)C1 N1(C(c2c(CC)ccs2)=O)CCC2C(CCCN2C(=O)CCc2cnccn2)C1 N1(C(c2c(C)nsc2N)=O)CCOCC(C(=O)NC(C)CN(C)C)C1 CC(C)CC(CNC(c1cccc(I)c1)=O)NC(c1cnc[nH]1)=O Cc1cc2c(C(=O)NCC(C)(CO)NC(C34CCCC3C4(F)F)=O)cccc2[nH]1 C(=O)(CCS(C)=O)NC(C1(CNC(=O)C(c2ccc(Cl)cc2)(F)F)CC1)C CC1CN(C(C2CCCSS2)=O)CC1(C)CNC(=O)CC1CCC2CC2C1 C1(O)(CC#C)CCN(c2nnc(Cc3ccccc3)n2C(C2(C)CC2)C)CC1 c1(CNC(c2ccc(Br)cc2Cl)c2n(CCOC)nnn2)cccc2c1OCO2 c1(C(=O)NC(C)C(CO)NC(c2ccc(CF)cc2)=O)cccc(=O)n1C N1(C(c2ccccc2Br)C(=O)NC2CCCCC2)C2CCCC1CC(F)(F)C2 c1(C(=O)OC)csc(S(=O)(=O)N2CCC(CC(N)=O)CC2)c1 C(=O)(NN1CC(C(N(C(CC2CC2)C2CC2)C(C)C)=O)CC1=O)OCC N1(C(C#CC(C)C)=O)C(CNC(C2CCC3(C2)CC3(F)F)=O)CC2CCCCC12 Cc1nc2c(N3CCOC(CC(N4CCNC(=O)C4)=O)C3)ncnc2[nH]1 C1(CC(=O)N(C(CNC(Cc2cn(CC)nn2)=O)C)C)C(=O)NN=C1C CC(C)CCCC(=O)NC(c1ccccc1)CNC(C1(C)CCC2CC2C1)=O N1(C(C(C)C2CC2)=O)CCC(N(C(=O)CC(c2ccc(F)cc2)O)CCO)CC1 c1(CC(C)C)cc(C(=O)NCC2CC2NC(=O)C(C(C)C)NC(N)=O)n(C)n1 C1(C(=O)NC(C)(CNC(c2ccsc2C(F)(F)F)=O)C2CC2)CC2OC1C1CC21 Cc1nnc2n1CCC(C(=O)NC1CCC(NC(=O)CC3COC4CC3C4)C1)C2 c1(SC)cc(C(=O)N(C)CCOCCN(C)C(C2CN(C3COC3)C2)=O)ccn1 c1(SCC(C)C)cccc(C(=O)NCCC(O)CNC(C2(O)CCSC2)=O)c1 c1(C(N2CCCC(NC(C(C(C)C)NC=O)=O)C2)=O)cc2c(s1)CSC2 c1(C(=O)NCC2C(NC(CNC(CC)=O)=O)CCC2)c[nH]c2cc(F)ccc12 c1(OC)ccc(NC(c2sc(-c3ccccn3)nc2C)=O)cc1[N+](=O)[O-] C1(C(=O)NCC(C)(C2CC2)NC(c2cnc(Cl)[nH]2)=O)CN2CC3CC2(CO1)C3 C1(CNC(COCC=C)=O)COCCN(C(=O)CCCCCC)C1 N1(C(C23C(CN(C(c4ccc(O)nc4)=O)C2)CC3)=O)Cc2cc(O)nnc2C1 C1(C(=O)NCCOC)CCC12CCN(C(c1cccc(NC3CCC3)c1)=O)CC2 N1(C(=O)CCc2ccccn2)CC2CC1CN2Cc1ccc(C(F)(F)F)cc1 C(CC(C(=O)N1CCCC(CF)C1)NC(C1C(C#N)C1(C)C)=O)OCC C(C(C)C(F)C(=O)NCCc1nc(C)no1)NC(C(CO)OC)=O C#CC1CC(NC(=O)C(C)=CCNC(=O)Cc2ccc(C)s2)C1 c1(C(=O)NCCC2CN(C(Cn3ncc(CC)c3)=O)C2)cccc(C(C)C)c1F C1(C)(CC)CC(NC(C2CC(C)(CC(=O)O)C2)=O)CCO1 c1(C(=O)NC(CC=C)CNC(=O)C(C)C2CCC2)ccc(Cl)c(C)c1 C1(OCCC)CCN(c2ccnc(NC3CCC3CO)n2)CC1 N1(C(COCCC=C)=O)CC(NC(c2cccc(=S)n2O)=O)CCC1C C(C)(CO)(C(=O)NCC1CCCN(C(C2CC(Cl)(Cl)C2)=O)C1)NC(C)=O CC(C)CC(C)CC(=O)N1CC2CN(C(=O)Cn3cccnc3=O)CCC12 CC(C)CCC(O)C(=O)NC(Cc1ccc(Cl)cc1Cl)C(=O)NCC(C)N=[N+]=[N-] Cc1cc(C(=O)NC(C)(C)CCC(=O)N2CCOC(C)(C(N)=O)C2)cc(C)n1 c1(OC)cc(C(N2CC3(CCCN3C(=O)CS(C)(=O)=O)C2)=O)cc(F)c1F Cc1cc(C(F)F)oc1C(N1CCCCC1CNC(=O)C(C)Cc1cnco1)=O c1(CC)nc2c(C(=O)NC3CC(C)N(C(=O)CCC[N+](=O)[O-])C3)ccnc2[nH]1 n1(CC(=O)NC(C)CCO)ccc2ccc(-c3cccc(C(C)(C)C)c3)cc12 C(=O)(C1=NNC(=O)CC1)NC1(C)CC(NC(c2cn(CC)nc2C(F)(F)F)=O)C1 c1(OC)ccc(C(N2CCNC(C(=O)NCCn3cccc3C=O)C2)=O)cc1O c1(C(N(C2CCCN(C(=O)NCC3CC3)C2)C)=O)ccc(NC(N)=O)cc1 c1(CC)cc(C(=O)N(C2(CC(=O)Nc3ccccc3C)CC2)CC)n(C)n1 c1(C(N2CCC(CCC(=O)NC(C(=O)OC)CO)CC2)=O)cc(C)cc(O)n1 N1(C(c2cc(C)on2)=O)CCCC(C2CCCCN2C(=O)CC2(CO)CCC2)C1 n1(CC(=O)N(C2CCCN(C(=O)CC(C)C)C2)CC)ccc2c(N)cccc12 c1(OCC)nscc1C(=O)NCCN(C(C1C(C)CC1C)=O)Cc1ccccc1 Cn1ccnc1-n1cc(CNC2(CO)CCO2)nn1 N1(C(C(C)OCOC)=O)CC(C)(N(C(=O)Cc2cc(C)[nH]n2)C2CC2)C1 C1(CCNC(CN(C(=O)COc2ccccc2)C)=O)CCCN(C(=O)C2CC2)C1 CCCC(C)CC(=O)N1CC(NC(=O)C=C(C)I)CC1(CC)CC C(C(C(F)(F)F)OCc1ccccc1)N(C(C(=C)C)C)CC N1(C(C)C(=O)NCc2ccc(CO)cc2F)C(=O)c2ccccc2C1=O c1(CC)nc(=N)[nH]cc1C(=O)NCC1CCN(C(=O)CCC2CCCN2C)C1 N1(C(C2(CC#C)CCC2)=O)CC2CN(C(=O)CC3CCCS3(=O)=O)CC2(C)C1 C=CCCC(F)(F)C(=O)NCC1(CCNC(C2CN3CCCN2CC3)=O)CC1 C(=O)(C(C)(C)C(O)C(C)C)NC(COC)CC(=O)Nc1ccc(C)nc1 C1(C(N2C(CNC(COCc3ncc(C)o3)=O)CCC2)=O)COCCC1(F)F c1(C(N2C(C(=O)NCCCC=C)CSCC2)=O)cccn2cncc12 N1(C(CC(=O)OCC)=O)CCCC2(CCCCN2C(=O)C(c2ccc(C)o2)C)C1 CCC(C)(C)C(C(=O)NCc1cccc(NC(=O)COC(C)=O)c1)OC C(CCCOC)(C(=O)NCC)ONC(C1CC=CCC1)=O.C=CC C1(CC(=O)NCc2c(C(=O)NCCC3CC(C)C3)c[nH]n2)CCCC12CC2 c1(C(=O)NCC(C)(C2CC2)NC(C2C(F)(F)C23CC3)=O)ccc([N+](=O)[O-])cc1N c1(C(=O)NCCC(C)NC(C2CC(=C)C2)=O)ccc(-c2ccnn2C)cc1 C1(C(=O)NCCCCCC=C)CCN(C(C2COCCN2C)=O)C12CCC2 N1(C(C(C)NS(CC)(=O)=O)=O)CCN(C(C2CC3C=CCC(C2)C3)=O)CC(O)C1 c1(CC(=O)NC(CC)CNC(=O)CNC(c2cccs2)=O)c[nH]nc1O c1(COC)csc(C(N2CC(CC(C)NC(=O)Cn3cc(C4CC4)cn3)C2)=O)c1 C1(C(=O)Nc2c(C)scc2)N(C(C2OCCCC2(C)C)=O)CC12CCCC2 N1(C(C2(C)CCC(=O)C2)=O)CCCCC12CC(NC(=O)CN1CCSCC1)C2 CC(C)C(C)(O)C(=O)NCC1CCN(CC(Cc2ccccc2)OC)C1 Cc1cc(C(=O)NCC2(F)CC(NC(c3cncc(F)c3)=O)C2)ccc1C1CC1 N1(C(Cn2cc(C(C)O)nn2)=O)Cc2ccccc2C(NC(=O)Cn2cncn2)C1 c1(N2CC=C(C)CC2)nc(C)nc(-n2ccc(C)n2)c1C CC(C)CCCCC(=O)NCC(O)CCNC(c1c(C2CCC2)cnn1C)=O C#CC(C)(C)C(=O)NCC(O)CN(C)C(c1cnncc1C(F)(F)F)=O Cn1cc(C(N2CCC(C)(NC(=O)CC3CCNC3=O)C2)=O)c(-c2cccs2)n1 CC1CN(C(=O)CC2CC(C3CC3)C2)CCN(C(c2cocn2)=O)C1 c1(CC(=O)NCCN(C(=O)C(N)=O)CCC)csc(C(C)C)n1 Cc1ccc(C(N2CCN(C)C(CNC(C3CCCN3C=O)=O)C2)=O)c(N)c1F c1(C(N2CCC3C(C2)CN3C(=O)CC2=CCCCC2)=O)cnc2c(c1)CCCC2 N1(C(C(COC)(C)O)=O)CCC2(CCCN2C(c2cc(C)c(F)cn2)=O)C1 c1(COC(CC(c2ccc(CC)cc2)C)=O)nc2ncccc2o1 N1(C(C(CC(F)F)N(C(=O)COc2ccsc2)C)=O)CCc2cncnc2C1 N1(C(c2c(C)nc(O)[nH]2)=O)CCCC2(NC(=O)COCC(F)F)CCCC12 C12(CNC(C(C)NC=O)=O)CC(CO1)N(C(=O)C(C)CNC(N)=O)C2 N1(C(CC(C(C)C)O)=O)CC2(C=C(C(=O)N(C)CC3COC(=O)N3)CO2)C1 c1(-c2cc(CC)[nH]n2)nc(C2CCCC3CC23)n(C2CCc3ccccc32)n1 c1(CCC(=O)NC(C(C)NC(=O)C=Cc2cscn2)C)ccc(Cl)nc1 N1(C(C(C)OCC=C)=O)CCC(CNC(=O)CCN2CCC2)(COC)C1 N1(C(C(Cn2ccc(C)n2)C)=O)CC2CC1CN2C(c1sc(=N)[nH]c1C)=O C(=O)(C(O)C1=CCCCC1)N1CCC(C(=O)NC(CCO)C(F)F)C12CCC2 C1(CNC(=O)CO)CCCCN1C(c1cc(-c2ccco2)on1)=O C(=O)(C(F)(F)C(F)F)NCC(CNC(c1c(C)nn(C(C)(C)C)c1)=O)O c1(C(=O)NCC(CN(C)C(c2coc(C(F)(F)F)c2)=O)O)cncn1C1CC1 N12CCC3CCN(C3C1)OCC2=O.C1(C(=O)OC)C=CC1C(=O)NC1CC=CC1 CC1CCCN(N=C2CCCNC3(CNS3)C2)C1C(=O)c1cnsn1 c1(C(N(CC2CCCN(C(C(CC)OC)=O)C2)CC)=O)c(OC)cccc1Cl c1(C(N2CCC(C(C)C)CC2)=O)ccc(S(=O)(=O)C2CC2)cc1.C1CS1.C(=O)OC C(c1ccncn1)=CC(=O)NCCCN(C(C1CCCN(C(N)=O)C1)=O)CC C(CC(C)(C)CC(=O)N1CCC2(NC(=O)CN3CC4C=CC3C4)CCCC12)OC N1(N(C(c2sncc2Br)C(=O)NC(CC)C)C2CCOC2)CCOCC1 N1(C(C2(CC=C)CCCCC2)=O)CCCCC(NC(c2cnc3n2CCC3)=O)C1 c1(OC)ccc(C2CC2)c(C(N2CCOCC(NC(C3C(C)C3C)=O)C2)=O)c1 C(CCC(C)C(=O)N(C1CCCNCC1)Cc1ccccc1Br)OCC c1(C(=O)NC2CN(C(=O)C(O)C3CC3)CC23CC3)cc(=O)c2ccc(Cl)cc2o1 N1(C(C(CC)Br)=O)CCC(N(C)Cc2ccc(SC)s2)C(F)C1 C1(C(=O)NOCCF)CC12CCN(C(=O)Cc1ccc(F)cn1)CC2 N1(C(c2c(C)ncc(N)c2)=O)C2CCC1CC(CNC(c1c(C)noc1C)=O)C2 N1(C(COC(C)C)=O)CC2CCC(C1)N(C(=O)C=Cc1cn[nH]c1)C2 N#Cc1ccc(NC(C2C3CN(C(c4ccnc(Cl)c4Br)=O)CC23)=O)cc1C#N Cc1cccc(C(C2CCN(C)CC2)NCCCSCC(C)C)c1 N1(C(C(CCSC)O)=O)CCC(C)(C)C(CNC(=O)C(C)Cc2ccco2)C1 C(=O)(CCc1cn[nH]c1)NCCN(CCOC)C(C1CC1C(=O)C1CC1)=O C1(NC(C2(CC)CCN(C(=O)C(COC)N(C)C)C2)=O)CCN(C)CC1(C)C C(c1cncnc1O)=CC(=O)NCC1(O)CN(C(C2CC2F)=O)C1 c1(C(N2CCC(O)C(C)C2)C(=O)NCCSC)ccc([Si](C)(C)C)s1 CCC(C)C(C)C(=O)N1CCC(CN(C)C(c2ccsc2C(=O)OCC)=O)CC1 C12(C(N(CCCN(C(=O)CCc3cncc(F)c3)C)C)=O)CC(C#N)(C1)C2 c1(C(=O)NC(CNC(CCSCC)=O)C(C)C(C)C)cc(S(N)(=O)=O)n(C)c1 c1(C(=O)NC(CCSC)C(=O)Nc2cccnc2)cc(C)cc(C)c1 c1(NC(c2nccn2-c2cccc(F)c2)=O)ccnc2cc(Br)ccc12 C1(C(N2CC(NC(C3C(CCOC)C3)=O)C2)=O)CC12CCCCC2 C1(C(N2CCCC(OCC)C2)=O)CN(C(=O)C(=O)C2CC2)CCC1O c1(C(C(=O)NC(CC)CNC(c2cn(C)c(O)n2)=O)C)ccc(F)c(F)c1 CN1CC2CC1CN2C(=O)CCN(C(=O)C(C)(C)CN(C)C)C1CC1 C(=O)(C(F)(F)C(C)O)NCc1c(CNC(c2nc(CS(C)(=O)=O)sc2)=O)ocn1 N1(C(C2OCC(C)(C)OC2)=O)CCC2C(CCCN2C(c2cnc[nH]2)=O)C1 c1(C(N(CCNC(C2(C)CNC(=O)C2)=O)CC)=O)ccc(F)c(S(C)(=O)=O)c1 Cc1ccc(Br)c(C(N2CCCC(NC(=O)CCOc3cccnc3)C2)=O)c1F N1(C(CCCCNC(c2ccc(C)nc2)=O)=O)CCN(C)CC1CCO CC1(C)OCCCC1CCN1CCCC1Cc1cn(CC2CCC2)nn1 Cc1ccc(C(N2CCC(CNC(=O)CC3CNC(=O)C3)CC2)=O)cc1C#N C1(C(N2CCC(CNC(CC(C)C3CC3)=O)C2)=O)COCCN1C(c1ccco1)=O Cc1cc(Cl)ccc1CC(=O)NC1CC12CC(NC(c1occc1C)=O)C2 c1(CC)cc(C(N2CC(CNC(c3ccc(Cl)nc3N)=O)C(C)C2)=O)ccc1F N1(C(C(C)C(C)O)=O)CCC(O)(C2CCN(C(c3cn(C)cn3)=O)CC2)CC1 N1(C(Cc2c(C)n(C)nc2)=O)CCC(NC(C2(C3CCCO3)CC2)=O)C(F)C1 Cn1nnc2cc(C(=O)NC3COCCC3NC(c3ccccc3O)=O)ccc12 c1(N2C(C(N3CCOCC3CO)=O)CC(C)C2)ccc(C2=CCSCC2)nc1 C1(C(=O)NCc2occ(C(=O)NC(c3ccncc3)CC)c2)CCC(=O)N(C)C1 CC(=O)CC(C)(C)C(=O)NC(C)CNC(c1ocnc1C(F)F)=O N1(C(c2cnn(C)c2F)=O)CCC2C1CCCN2C(c1cc(C(C)(C)C)on1)=O C1(CNC(C2(CC(C)C)CC2)=O)CCCC2(CCN(C(=O)CC(C)C(C)C)CC2)O1 C1(CNC(C(CC(C)C)O)=O)CCC2(CCN(C(=O)C=CCO)CC2)O1 Cc1c(CN2CCOCC(C(=O)N(C)Cc3cnn(C)c3)C2)cccc1[N+](=O)[O-] c1(C(N2C(CNC(C3CC(OC)C34CCC4)=O)CCC2)=O)cn(C)c(=O)nc1O C1(C(N2CC(OCC)(CNC(c3ccc(CO)cc3)=O)C2)=O)CCC12CCCO2 CC1CCC(C(=O)N(CCCCCNC(c2scnc2C(F)(F)F)=O)C)C1 CC(C)CC(C(=O)NC(C(=O)NCC1CC2(CCC2)C1)C1(O)CCC1)C(N)=O C(=O)(CCN(OC)C(=O)C=Cc1cnn(C)c1)N(C(CS(CC)(=O)=O)C)C Cc1cc(C(N2CCC(NC(=O)CC3CCC3C)CC2)=O)c(F)cc1F N1(C(CS(N)(=O)=O)=O)CC2(COC(CNC(c3cc(C4CCCC4)[nH]n3)=O)C2)C1 c1(C(C(=O)NCC(CC=C)NC(C23COCC(C2)C3)=O)CO)ccc(Cl)cc1 c1(SCC#C)ccc(NC(=O)Nc2nccn2CC2CCCO2)cc1 C1(CNC(CCOC)=O)CCCC2CN(C(C3CC4CCC3C4OC)=O)CC12 C(C)(C(C)C(=O)Nn1cnn(C)c1=S)NC(CSCC)=O c1(CNC(C(CC)C)C)cc(F)c(N2CCOCC2)c(F)c1 CN1C(=O)c2ccccc2C1C(=O)NCC1(O)CCN(C(=O)CC2CCCC2)C1 N1(C(C2C3(CCN(C(Cc4n(C)ncn4)=O)CC3)C2)=O)CCc2c(cnn2C)C1 Cn1cc2ccc(C(=O)NC34CCN(C(C5(C)CC=CC5)=O)CC3C4)cc2n1 C1(CC)CCCCC1OCC(N1CC(NC(=O)CNS(C)(=O)=O)CC1C)=O CCCC(C#N)C(=O)NC1CCCC1NC(c1ccnc(S)c1)=O C(=O)(C(F)CC(C)C)NC(CC)CNC(=O)CCCc1ccc(C(C)(C)C)cc1 Cc1nc(O)ccc1C(=O)NCC(O)CC(=O)NC(c1ccccc1)C c1(C(=O)NC(C2CCCC2)CNC(c2cccs2)=O)c[nH]nc1-c1ccsc1 c1(OCC(=O)NCCC2(NC(CN(C3CCSC3)C)=O)CC2)ccccc1 CCCC(C(=O)NCC(C)NC(C1CCSCC1)=O)S(N)(=O)=O c1(C(=O)NC(=O)OC)cc(C)nnc1N(C1CCC1)C(C)C c1(C(=O)NC2CCCC(NC(c3ncccn3)=O)C2)cc2ccc(Br)cc2s1 C1(CC)CN(C(=O)C=Cc2ccco2)CCC1NC(C1CC2(CCC2)C1)=O C1(NC(=O)C2=NOCC2)CN(C(=O)COc2ccc(F)cc2)C2(CCOCC2)C1 C1(CNC(c2cc(Cl)n[nH]2)=O)(CO)CCCN(C(=O)COCC2CCCO2)C1 c1(CCC)ccc(C(=O)NC2CCN(C(C3CC(C(F)F)C3)=O)C2)cc1 CCCCCC(C)C(=O)N1CCCC(Nc2cc(COC)ncn2)CC1 C1(NC(C(n2ncc(C)c2)C)=O)CC2CCC1N(C(c1cc[nH]c(=N)c1)=O)C2 c1(NC(=O)NC(c2ccco2)CC)ccccc1SC(C)(C)CC C1(C(N2CCC(C(C)NC(=O)Cc3cnccn3)C2)=O)CCCC(F)C1 C(=O)(C(C(C)C)N1CCCCC1)NCC1CN(C(C=C(C)C(F)F)=O)C1 c1(C(=O)NC(C)CCN(C(=O)C(CO)NC(N)=O)C)cc(C(N)=O)cc(F)c1 c1(C(=O)NCC2N(C(c3c(F)cccc3Cl)C)CC2)n[nH]c2c1CCCC2 c1(N2CC(CC#N)N(C(=O)C=Cc3ccc(I)o3)CC2)ncnc2n[nH]cc12 c1(SC(c2cccc(SCC(=O)OC)c2)C)nc2ccc(Cl)cc2s1 C(C(CCN)NCCCN(C)Cc1ccccc1)OC C(=O)(C(CC(=C)C)NC(=O)C(CC)N(C)C)N1CCC(C=C)C1 CCC(C#N)C(=O)C(=O)CC1C2CNCC12.C(CCCCc1cnc[nH]1)N c1(C(=O)NCCCC2N(C(=O)OC(C)(C)C)CCC2)ccc2c(Cl)n[nH]c2c1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCCC(C2(NC(c3nnc(C)s3)=O)CC2)C1 O(P(=O)(CCC1CCN1C(=O)C(=O)NCCOc1ccc(F)c(C)c1)OCC)CC CC12CN(C(=O)COc3ccccc3Br)CC1CN(C(C1CC1Cl)=O)C2 C1(NC(=O)Nc2ccccc2OC2CC2)CCN(c2cc(C)c(I)cn2)CC1O N1(C(C(C(C)CC)NC(c2c(CC)non2)=O)=O)CC2(CCC1CO)CC2 c1(-n2cc(CN(C(c3c(C)cc(Cl)nc3N)=O)C)nn2)cc([N+](=O)[O-])ccc1Cl C(CNC(=O)C(F)OC(F)(F)F)(CCOC)NC(C1(OC)CCC1)=O C(CCOC)(C(=O)NC1(C(O)CO)CC1)NC(C(CC)=CC)=O C#Cc1nc(C(=O)NCCN(C(=O)CN(C)C)C2CC2)cs1 Cc1c(N(C2(CC(=O)O)CC3(C(=O)O)CCN3C2)C2CC2)cccc1C#N C(=O)(C(O)CC(F)(F)F)NCC(C)CC(=O)NC1(C)CC(F)C1 C1(C(C)(C)NC(C23CCC2C3)=O)CCCN1C(C1CC1Sc1ccccc1)=O C1(Cl)(C(=O)NCC(c2ccccc2)N(C(CN(CCC)C)=O)C)CC1(C)C Cc1c(C(=O)NC(C)C(C(C)C)NC(=O)Cc2ccsn2)ccn1CCO CCCCC(F)C(=O)N1CCCCC1CN(C)C(c1cc(C)[nH]n1)=O c1(C(N2CCCC=C2Br)=O)ccc2nncn2c1 N1(C(c2n[nH]cc2[N+](=O)[O-])=O)CCC2C(CCCN2C(=O)C=Cc2cc[nH]c2)C1 c1(NCC2CCC(CCC(=O)OC)O2)cccc2cc(OC)c(OC)cc12 N1(OC(CSCC(=O)NC(c2c(OC)cccc2)CF)=O)CC(C)OC(C)C1 Cc1cc(=NCc2c[nH]nc2C(C)(C)C)[nH]c(N2CCC(C)S(=O)(=O)CC2)n1 N1(C(COCCNC(c2nnc(O)nc2O)=O)=O)CC2(CCC(O)CC2)C1 C1(NC(CCCC(CC)C)=O)CCN(C(c2cnc(S)[nH]2)=O)CC(C)(C)C1 C1(NC(C(C(C)C)NS(C)(=O)=O)=O)CCC2(CC1)CN(C(c1cnnn1C)=O)C2 CC(C)CCCC(=O)N1CC2(NC(c3nn(C)nc3C(=O)OC)=O)CC1C2 N1(C(C(COC)(C)C)=O)C2CCCC1CN(C(C1Cc3cccc(C)c3O1)=O)C2 C1(CN(C)C(C2CCS(=O)(=O)N2)=O)CCCN(C(=O)CN2CC(F)(F)C2)C1 C1(CNC(C2N(S(C)(=O)=O)CCCC2)=O)COCCN(C(C2(N(C)C)CC2)=O)C1 C1(C(=O)NC(c2cccnc2)C(C)C)C2CC1N(C(c1ccncc1F)=O)C2 c12ccc(cc1F)c(=O)[nH]2.C1(NC(C)=O)(CO)CN(C(c2cc(CO)no2)=O)C1 C=CC(CC(=O)NCC1CCC1NC(=O)C1=CCSC1)c1ccc(OC)cc1 N1(C(CC=C)=O)CCCC(C2(NC(c3n[nH]c(C)c3Br)=O)CC2)C1 S(=O)(=O)(c1ccc(Br)cc1NCC1CC2(CCOC2)C1)NCC(C(C)(F)F)(C)C C1(C)(C(N2CC3(N(C(CC4(OC)CCOCC4)=O)CC3)C2)=O)CC(C(C)C)=NO1 C(c1ccccc1Cl)=CC(=O)NC1CN(C(c2cc(F)ncc2Br)=O)CC1F c1(CN(C(=O)OC(C)(C)C)C2CC2)ccccc1-c1noc(CCC(N)=O)n1 C1(C(=O)NC2(C)CN(c3nc(Cl)c(C#N)s3)C2)CC2CCCCN2C1 C1(OC(C)(C)C)CCCN(c2cncc(NC3CCN(C(N)=O)CC3)n2)C1 Cc1nc(CNC(C2(F)CC2)=O)oc1C(N1CC(c2ccccc2F)(F)C1)=O C(CCC(C)(C)C(=O)N1CC=CC(NC(=O)C(C2CCCCCC2)C)C1)OC c1(C(N(C2CCN(CC)C2)C)=O)cc(O)n(CC)n1 C12(NC(c3cnn(C(C)C)c3Cl)=O)CCCN(C(C3CCCC(=O)C3)=O)CC1C2 c1(OCC(=O)NCCC2CN(C(C3(C)CC3)=O)CC(C)O2)cccc([N+](=O)[O-])c1 N1(C(Cc2c(C)noc2C)=O)CC2CCN(C(C3CCCCC3(F)F)=O)CC2C1 N1(C(C(C)n2ccnc2)=O)CCCN(C(c2cccc(C(F)F)c2F)=O)C(C)C1 C(=O)(CC(C)(C)CC(F)(F)F)N(C1CCN(C(C(CC)(C)C(N)=O)=O)C1)C c1(CC)c(C(=O)NCC2CN(C(=O)CC(C)F)C(C)(C)C2)sc2ccccc12 C1(CC(=O)NC(C2CCOCC2)C)CN(C(C2CCCC(=O)C2)=O)CCC1C C12(C(=O)NCc3cnc(C)o3)C(NC(=O)CCC3CC3(F)F)C3CC1C2C3 CCC(CC(=O)NCC(CC(=O)NCC1(O)CCN(C)C1)C1CCC1)C(C)(C)C C1(C(=O)NCC2N(Cc3cn(C)nc3C3CCC3)CC2)CCCCC1(F)F N1(C(c2cncc(C(F)(F)F)c2)=O)CCC2(CCCC2)C1 N1(C(C2N(CC)CCCC2)=O)CC2C3CCC(C3)C2C1 C=CCC(C)(C)C(=O)N1CCC(C(C)C(=O)NCC(C)(CC)C(N)=O)CC1 c1(OC)ccc2sc(CN(C=O)C(c3ccc(OC)nn3)C)c(C)c2c1 C(CCC)(C(O)C(=O)N1CCCC1CN=[N+]=[N-])NC(C(C=C)O)=O Cc1nc2nccc(NC3CC(C)N(C(=O)C(C)(F)F)C3)n2n1 c1(C(N2CCC(C)C2C)=O)ccc2c(c1)CN(C(=O)N=c1cncc(CN)[nH]1)C2 N1(C(Cc2c(C)cccc2)=O)CCN(C(c2cc(CO)[nH]n2)=O)C(C)C1C N1(C(C(C)C)=O)CCC2CCC(NC(c3ccc(Cl)c(Cl)c3)=O)C1C2 C1(NC(c2c(C)n(C)nn2)=O)CCN(C(c2cc(Br)nn2C)=O)CC1F N1(C(C(=O)N(CCc2cn(C)nc2)C2CC2)=O)CCCCC1CCC1CCOC1 c1(C(N(C2CCN(C(C(COC)(C)C)=O)CC2)C)=O)cc(F)cc(F)c1 C1(OC(C2CC(OC(C)(C)C)C2)=O)CC2(C1)CN(C(=O)CC1NC(=O)NC1=O)C2 C1(NC(C(CCCCC)O)=O)CN(C(C23CCOC(C)(C2)C3)=O)CC2(CCC2)C1 CC1(C(N2CC(NC(=O)CCc3ccc(Cl)cc3)C(O)C2)=O)COCC1(F)F Cc1c(O)ccc(C(N2CC3CC(Nc4cccc(C#N)n4)C3C2)=O)c1C C12(F)CCCN(C1)C(=O)C1(CCCCC1)NC2=O.c1(COC)cccc(CO)c1 C(CCCC(C)NC(C1(OC)CCSCC1)=O)NC(C(CC1CC1)OC)=O c1(C(=O)NCC2CC(NC(C(c3cccc(Cl)c3)CC)=O)C2)cn(C)c(O)n1 C1(CNC(C(C(C)C)OCC)=O)CN(C(C2(CN(C)C)CCCC2)=O)CCN1C C(=O)(C(C)(C)C#N)NC(C1CCCN(C(=O)CCSc2ccccc2F)C1)C C1(O)(CNC(c2c(C)nc[nH]2)=O)CCN(C(=O)CC2OCCC2(C)C)C1 c1(C(N2CCOCC(NC(C=COCC)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 N1(C(c2cc(CC)oc2C)=O)CC2CC(C1)N(C(c1cc3sccc3s1)=O)C2 N1(C(CCCCOCC)=O)CCN(C(=O)C(C)N2CC(C)C2)CC12CCC2 CCCC(C)CCCC(=O)N1CCC(NC(c2oc(CCC)nc2C)=O)C1 C1(NC(C2CC(NC(CCCC=C)=O)C(O)C2)=O)CCCC(O)CC1 c1(C(=O)NCC2N(C(C(C)SCC)=O)CC2)cccc(F)n1 c1(C(N(C)CC2N(C(C(C)OCCC=C)=O)CC(F)C2)=O)cccc(N)c1Br N1(C(C#CC(=O)N(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2ncccn2)=O)C1 N1(C(=O)CSCc2nc[nH]n2)CC2(CC(CO)C2)C1.C12(C(=O)N)CCC(CO)(CC1)C2 C(c1cccc(O)c1)=CC(=O)NCC1CCCN(C(C2C(C)=CCC=C2)=O)C1 C1(O)(CCNC(C(C)N2CCC2)=O)CN(C(=O)C=C2CCC(C)C2)C1 N1(C(C(C)CC#N)=O)C2CCC(C2)C1C(=O)NCCN1CCC(O)C1 CCS(=O)(=O)C=CC(=O)N1CC(F)(F)CC1CNC(=O)C(F)Cc1ccccc1 N1(C(CCCOCC)=O)CCN(C(=O)C(C)N2CCC2)CC1c1cccnc1 C1(C(=O)NC(CN(C(C(C)OCCOCC)=O)C)C)CCC(=C(F)F)CC1 Cc1ccc(OCCC(=O)N(C)CC2CCN(C(=O)C=CC3CC3)CC2)cc1C c1(C(=O)NCC2(NC(c3ccc(C(F)F)cc3F)=O)CC2)ccc(O)c(F)c1 c1(C(=O)NC(C(C)C)CNC(C2CC2C)=O)cc2cccnc2cc1F c1(NC)ccc(C(=O)NC2CC2CNC(=O)COc2ccc(COC)cc2)cc1 N(C(=NCCF)N1CCCC2(CC2)C1)CCN1CC(F)(C(C)(C)CNC(N)=O)C1 c1(CC(C)C)nn(C)cc1C(=O)NC1CCN(C(=O)CC2CC(=O)NC2=O)C1C CC1(C(N2CC(NC(c3nccc(C(F)F)n3)=O)C2)=O)CC(C2CC2)=NO1 C(=O)(C1c2ccccc2OCC1(C)C)N1C(CNC(c2ncc(C)c(Cl)c2)=O)CC1 N1(C(c2ccc(OCC(C)C)cc2)=O)CCN(C(=O)C(O)C(F)F)CC(C)(C)C1 C12CCCN(C1)C2=O.n1(C(C(=O)NC(C)C)C)cc(-c2cc(C(N)=O)cs2)nn1 CC1CCCC(C(=O)NCC2CCN2C(=O)Cc2ccnc(C(F)(F)F)c2)C1 C1(NC(c2c(CC)c[nH]n2)=O)CCCC(N(C)C(C2CC(O)C2)=O)C1 c1(CC(=O)N(CCN(C(=O)C(C)(C)c2ccns2)C)C)cccc(C#N)c1 c1(C(N2CC(CNC(=O)CC3CCC(O)C3)OCCC2)=O)n[nH]c2c1CCSC2 N1(S(CC)(=O)=O)CCC2(CC1)CC(C(CC)NC(=O)CSC(C)=O)C2 N1(C(C2(OCC)CCCC2)=O)CCC2(CCC(NC(C3(C)CC(F)C3)=O)C2)C1 CN1CCN(CCC(=O)N(CCCNC(C2CCC(O)C2)=O)C)CC1 CS(=O)(=O)C(CN=c1[nH]c(N2CC3CCC3C2)nc2c1SCC2)C1CC1 C1(NC(CO)CSc2ccccc2)CNCCOC1 CON1CCC(C(=O)NC2CN(C(c3cn(CC(F)F)cn3)=O)CC2F)CC1 N1(C(=O)CNC(=O)C(C)NC(C)=O)CCCC(NC)C1.CCCCNC(=O)CS C1(C2CC2)(NC(CCNC(CC(C)C)=O)=O)CCCC1 CC1CC(NC(=O)CN2CCS(=O)(=O)CC2)CCN1C(c1nncs1)=O c1(C(N(C2CCCC2)CCCNC(C(=O)NCC)=O)=O)c(C)nc2sccn12 c1(NCCc2c(C)cccn2)cc(Br)ccc1S(=O)(=O)N1CCN(C=O)CC1 N1(C(CCCCCOCC)=O)CCC2(CNC(C3(C)CC3(F)F)=O)CCCC12 c1(CC)nc(C(=O)NCC(O)CC(=O)NCC2CCCOC2)c(C)o1 CCCC(CC)C(=O)NC(CCC1CC1)C(=O)NCCN1CCCCC1=O c1(C(=O)NC2CCCN(C(C=CCC)=O)CC2)ccccc1S(C)(=O)=O C1(C(=O)NCCOCC#C)CN(C(=O)C=CC)CC12CC2 c1(CCC)ccc(N)c(C(=O)NC2CCCC2NC(=O)C=CC2CCOCC2)c1 C1(C(N(CCCCCNC(C2C(Cl)(C(=O)OC)C2)=O)C)=O)CC2C=CCC(C1)C2 C1(CC#C)(C(N2CCC(C(C)NC(=O)C(F)C3CCOC3)C2)=O)CCOCC1 C1(Nc2ncc(Br)nc2)CCn2nccc2C1 N1(C(=O)NCC(COC)C)CC2COCC2(C(N2CCCC(OC)C2)=O)C1 c1(OC)nccc(C(=O)NC2CC(CC(=O)NCC(C)O)C2)n1 c1(C(N(CCNC(C2C(C(C)C)CCO2)=O)C)=O)cnc(Br)c(N)c1 CC1=CCC(C)(C(N2CC3C(CNC(c4cnn(C5CC5)c4)=O)C3C2)=O)CC1 C1(N(C)C(c2cc(Cl)no2)=O)CC2CC1N(C(=O)CCc1ccc(F)cc1)C2 N1(C(CCN(C2CC2)CC)=O)CC(O)CC1(C)C(=O)NCc1nccn1CC N1(C(=O)OC(C)(C)C)CCC(NCc2ccc(Br)cc2)C(C2CCOC2)C1 CCCCC(C)(F)C(=O)NCC1C2CN(c3cc(C(F)(F)F)nc(C)n3)CC12 CCC(=O)CCC(=O)N1CCOCCC1C(=O)NCC(c1ccccn1)O N1(C(CCc2onc(C)n2)=O)CCCCC(C2CN(CC3CC(F)(F)C3)C2)C1 C#Cc1cccc(CC(N2CCCCC2CNC(=O)C(C)(F)CCC)=O)c1 c1(C(N2CC3CC(NC(C4CC=CC4)=O)CC3C2)=O)cnnc2ccccc12 N1(C(CCCN(C(=O)CCC(=O)C2CC2)C)=O)CCCNC(=O)C1 N1(C(c2cc(C)c(Cl)s2)=O)C2CC=C(C(=O)N3CCC(O)(C(C)C)C3)C1CC2 C(c1cccnc1)=CC(=O)NCC(N1CC(CC(C)NC(c2cccs2)=O)C1)=O c1(C(=O)NC23CC(NC(C=C4CCC(C)CC4)=O)(C2)C3)cnc2c(c1)CCC2 N1(C(C(C)OCC=C)=O)C2CCC1CC(NCc1ccnc(OCC)c1)C2 c1(C(C(=O)Nc2ccc(F)cc2)N(C(CC)COC)C)cnn(C)c1Cl C1(NC(C(CC(=C)C)C)=O)C(C)CC2CN(C(C)=O)CC12 Cc1c(C(N2CCOC(C(C)NC(=O)C3=CC(C)(C)C3)C2)=O)cncc1Br C1(N(C(C(CC)O)=O)CC(C)C)CCN(C(C2CN(C(N)=O)C2)=O)CC1 C1(NC(c2ccc3c(c2)CC3)=O)CN(C(=O)COCC2CCOC2)CCC1F c1(OC)ccsc1C(=O)N(C1CC1)Cc1cccnc1.C1(C)C=CC(=O)N1 C1(C)(C(=O)NCC2OCCN(C(C(C(C)C)N(C)C)=O)C2)CC(C(C)C)=NO1 C#Cc1cccc(C(=O)NCC2CC2CNC(c2ccccc2CCC)=O)c1 N12CCCCC1C2.C1(N(C(=O)C(Br)=C(C)C)CC)CCN(C(CC)CO)CC1 C1(C(N2CC(O)(CNC(=O)CCOc3ccc(F)cc3)C2)=O)CC2C=CC1CC2 CCCCCC(=O)NCC1CN(C(C2CN(C(C)C)CCO2)=O)CCO1 c1(OC)ncnc(OC)c1C(=O)NCC(C)(C)CNC(=O)C=Cc1cn(C)nn1 c1(C(N2CCCC(CCNC(C34COCC3C4)=O)C2)=O)ccc2occc2c1 c1(C(c2n(CC(=C)C)nnn2)NC)nc(C)sc1C.C1(C(N)=O)(N)CC1 c1(C(c2ccccc2)Nc2nnn(CC(N)=O)n2)ccc(I)cc1 C(=O)(C1CCCc2nncn21)NC1(C)CCCN(C(c2c(CCC)nco2)=O)C1 Cc1nc(C(=O)NCC2(NC(=O)CSc3nccn3C)CCC2)c2ccnc-2[nH]1 c1(NC(C(CC2CC2)NC(=O)CCn2cncn2)=O)ccccc1Cl N1(C(c2c(OCC)nccc2)=O)CC2CC1CN2C(c1cn(C)c(=O)n1C)=O c1(CNc2cc(C)c(I)cc2)sc2cccnc2c1Br C(CC(C(C)(C)C)NC(c1ncnc(O)c1Cl)=O)N(C(C(CC)(C)O)=O)C N1(C(C(CC)Oc2ccccc2)=O)CC2CC2(C(=O)OCc2[nH]nnc2OC)C1 c1(N2CCCC(OC)C2)ccn2ncc(S(=O)(=O)NC3CC(O)C3(C)C)c2n1 N1(C(C2(OC)CCC2)=O)CCC(O)(CCNC(C2CC2C(C)C)=O)C1 C(C(C)C(C)C(=O)NC1(CF)CN(C(=O)C(C2CCCN(C)C2)(C)C)C1)OC N1(C(Cc2c(C)nccc2)=O)CCC(C)C(NC(=O)CCC2CCCCC2)C1 C1(C(N(CC(C)(C)NC(c2c[nH]nc2C2CC2)=O)C)=O)CCCCC(F)(F)C1 C1(CC(=O)N(C)CC2N(C(COCC(=O)NC)=O)CCC2)CCOC1(C)C N1(C(=O)C=Cc2nccs2)CCN(CC2CN(C(=O)CC3CCCCO3)C2)CC1 N1(C(CC2(CC)CCC2)=O)CCOCC(CNC(c2cnn(C3CC3)c2C)=O)C1 C(C(C)C)(C(O)C(=O)N1CCCCC1CNC(=O)C(C)SC)OC CCCCC(C)(F)C(=O)NC1CC2CC(C1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 N1(C(CN(CCOC)C)=O)CC2CCC1CN2Cc1cc(NS(C)(=O)=O)no1 C1(NCC2(O)CCC(C)C2)(NC(=O)OC(C)(C)C)CCc2cc(Br)ccc2C1 C(C)(CNC(C1CC(C(F)(F)F)(OC)C1)=O)(C(C)C)NC(CC1CC(=C)C1)=O C1(C)(CNC(C(C)N(C(=O)C=CC2CCCCC2)C)=O)CCC(=O)N1C CC1=C(C(=O)N2CCN(C(C3(n4cccn4)CCOCC3)=O)CC2)CCO1 c1(CC)cc(C)ccc1C(=O)N(CCN(C(=O)C(C1CC1)OC)CC)CC c1(NC2C(COC)CCC2)cc(C(=O)NC2(CO)CCCC2)ncn1 c1(OC)ccc(C(=O)NC2CCC(N(C(=O)CSCC3(F)CC3)C)C2)nn1 N1(C(c2ccc(-c3n(C)ncn3)cc2)=O)CCCC(NC(=O)CC(F)(F)F)C(F)C1 c1(C(=O)NCCNC(C2(C)CCSCC2)=O)ccn2ccnc2c1 C(CCCCC(=O)N1CC(COC)CC1CNC(c1cccc(Cl)c1)=O)=CC C1(C(=O)NC(C(=O)NCC(C)C(C)(C)C)CCF)CC2(CCC2O)C1 Nc1cc(C(=O)Nc2cccc(CCNC(C3CC3C(=O)N)=O)c2)ccc1Cl c1(C(=O)NCCCNC(c2c(C)n(CCO)cc2)=O)nc(Cl)c(Cl)c(N)c1Cl c1(C(=O)NCC(C)=CC(=O)O)cccc(N2CCN(C)CC2)n1 CC1CCCn2c(C(N3CCN(C(C4CCC(C)(C)C4)=O)CC3C)=O)cnc21 C1(C(N2C(C)(C)C(NC(=O)C=CC(F)(F)F)CC2)=O)COC2(CCC2)CO1 c1(C(=O)NC2CC(NC(C3CCC(C)S3)=O)C2)[nH]c(=N)sc1C(F)(F)F C1C(C)(C)CC(=O)N2CC(O)CC2(C)C(=O)N1.C1(N(C)CC)CC(CSC)C1 c1(C2N(C(C(CCO)NC(=O)OC(C)(C)C)=O)CCC2)ccc2c(c1)OCO2 Cc1nc(CO)sc1C(=O)NC1CCOCC1NC(=O)C=Cc1ccncc1 CC1CN(C(=O)C(=O)NC2CC2)CC1C(=O)NCc1ccc(-c2csnn2)cc1 c1(C(N2CC(C(C)NC(c3ncccc3F)=O)OCC2)=O)cc([N+](=O)[O-])nn1C N1(C(c2ccc(C)n2C)=O)CC2OCC(NC(=O)C=Cc3cnn(C)c3)C2C1 N1(C(C(CCSC)O)=O)CCC(O)(CN(C(=O)C(C)CC(C)C)C)CC1 C(=O)(CCS(N)(=O)=O)NCC1C(CNC(C(C(C)C)n2cccc2)=O)C1 c1(CCC(=O)NCC(CN(C(C2C(OC)C2)=O)C)O)ccc2c(c1)NC(=O)CO2 CCCCCC(O)CC(=O)NC(C)CN(C(=O)CC1CCCCC1C)C N1(C(C(n2c(C)ncc2)C)=O)CC2(CNC(C3CCCC(F)C3)=O)CC(F)(C1)C2 C1(Oc2c(Cl)ncc(CC)c2)CCc2cc(OC)ccc2C1=O c1(C(=O)NCC2CC(NC(c3c(C(N)=O)cncc3)=O)C2)ccc([N+](=O)[O-])cn1 c1(OC)ccc2c(C(=O)NC3CCN(C(=O)Cc4ccco4)CC3F)csc2c1 c1(C(=O)NC(CC2CN(C(C(CC#C)O)=O)C2)C)ccc2ccn(C)c2c1 N1(C(c2ccc(SC(C)(C)C)s2)=O)CCC(NS(=O)(=O)NSC)C1C c1(C(N(C)C=O)=O)cccc(S(=O)(=O)NCC(C)N)c1 C(CS(=O)(=O)c1ccc(C)cc1)NC(c1cc(F)ccc1F)CC=C c1(OC)cc(C(N2CCN(C(=O)CCNC(C)=O)C3CC23)=O)cc2c1OC(C)C2 C(=O)(C1OCCc2ccccc21)NC1CC(NC(C=Cc2cn(C)nc2)=O)C1 c1(C(=O)NCCOCCCN(C(C(=O)NC(C)C)=O)C)nc2ncccn2n1 CN1C(=O)Cc2ccc(C(=O)NCC3(C)CCN(C(C4COC(=O)N4)=O)C3)cc21 N1(CC(=O)NCCOC)CC(NC(c2c[nH]cc2C)=O)C(C#N)C1 c1(C(N(C(C)C)CCNC(c2ccn(C)c2)=O)=O)ccc(Cl)c(Cl)c1N c1(CNC2C(C(=O)NC3(C(=O)OC)CCOC3)C2)cc(Br)ccc1C Cc1ccc(C(C(=O)NC(C(=O)O)c2cccs2)C2CC2)cc1 N1(C(C2CN(C(C)C)C2)=O)CCCC2CC3(CCC3)C12 c1(OC)cncc(C(N2CC(NC(C3CCOC3=O)=O)C(C)C2)=O)n1 c1(C(N2CCC(C)(NC(c3cccc(N)c3F)=O)C2)=O)cc2cc(F)ccc2s1 c1(CCCCc2cn(C(CNC(c3[nH]cc(CC)c3)=O)C)nn2)ccc(Cl)cc1 C(CC1CCC1)(C(=O)NCC(F)CO)NC(CSCCCC)=O Cc1conc1C(=O)NC(C(=O)N(CCCF)C)c1ccoc1 Cc1ccc(C(N2CC(NC(=O)C(C)(CO)CO)C(F)C2)=O)cc1F c1(CC)n[nH]c(=NCC2CCC(NC(=O)Cc3cccc(SCC)c3)C2)o1 C=CC(CCC)CC(=O)N1CCCC1CNC(=O)C=CCOc1cc(F)cc(F)c1 Cc1n[nH]cc1NC(c1nc(C(=O)NCc2ccoc2)cs1)=O C1(NC(CO)=O)(CSC)CCN(C(C2CCCN(C(N)=O)C2)=O)C1.C(CN(C)C)OC Cc1nc(C(N2CC=C(CNC(C3CSC3)=O)CC2)=O)ccc1C#N N1(C(CCN(CC=C)C(C2CC2(Cl)Cl)=O)=O)CC(F)CC(F)C1 N1(C(c2cc(OC)ncc2Br)=O)CCCC2(C1)CN(Cc1cccnc1)CCO2 C(=O)(C(CC1CCC1)Oc1ccc(C(F)(F)F)s1)NCC(OC)O N1(C(C2C(=C)C2)=O)CCCC2(CCN(C(c3ncoc3CC)=O)C2)C1 CC(CCNC(=O)C(=O)N(C)C)CCNC(C1=CN=CNC1C1CCNCC1)=O CC(C)(C)CC(C(=O)NOCc1nc[nH]n1)NC(C1CCN(C2CC2)C1)=O c1(C(=O)NC2C(C(=O)OC)CC2)nc(C)ns1 CCC(CC)CCCN(C)C(C1CSCN1C(=O)C=Cc1cc(C)no1)=O c1(NC(C2(C)CCCN(C(Cc3c(C)cccc3)=O)C2)=O)nc(Cl)c(Cl)cc1Cl C1(NC(c2cc(C)ns2)=O)CC2CC1CN(C(C1(C)CNC(=O)C1)=O)C2 C1(C(=O)NCCC2CC(NC(CNC(=O)OCC=C)=O)C2)CC2(CC2)C1 C12(C(=O)NC3(CC=C)CCC3)CC(CN1C(=O)CCCNC(=O)C(C)(C)C)C2 C(N=c1nc2ncn(C)c2c(NC2CCCC(C)C2)[nH]1)c1c(C(C)C)noc1 N(C(=NCCCN1CCOCC1)NC1CCC1)CCC1OCC(C(=O)OCC)C1 c1(CNC(=O)NCC(C2(C)CCCS2)(C)C)ccnnc1O C1(CCC(=O)NC(CC)C2CC2)CCCCN(C(=O)C(C)N(C)C)C1 C=C1CC(C)(NC(c2ccccc2)C2CCCC2)C1 Cc1cccc2c1CCN2C(=O)CC1CN(C(=O)CCCCC(=O)NC)CCC1C N1(C(c2c(CC)oc(C)c2)=O)CCC(CNC(c2cn3ccnc3s2)=O)C12CC2 c1(C(N2CC3CCC2CN(C2CC4(CNC4)C2)C3)=O)cc2cc(Br)cnc2[nH]1 c1(C(=O)OC)ccc(NC(c2cnn3c2CCC3)=O)c(F)c1F CC(C)(C(=O)NCC1CCCN1C(=O)C(C1CCC1)C1CCC1)N1CCCCC1 N1(C(C2CCN(C)CC2)=O)CC(NC(C2CSCN2C)=O)C(C2CC2)C1 c1(C(c2n(Cc3nnn(C)n3)nnn2)NC2CC(Cl)(Cl)C2)ccc2occc2c1 C1(C)(C(=O)NC(c2nncn2C)CC)CN(C(=O)CNC2CCCO2)C1 N1(C(C2N(C(C(SC)SC)=O)CCOC2)=O)C2C=CCC1CCC2 C1(NC(C2(C(F)(F)F)CCC2)=O)CCCC(NC(C2(C(F)F)CCCO2)=O)C1 c1(C(N(CCCCCNC(c2nn[nH]c2Cl)=O)C)=O)cc2nccn2c(O)n1 C1(CC(=O)NC(C(C)C)C2CCC2)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC1C c1(CC(=O)NCCC(C)(C)NC(C(C(C)(C)C)SC)=O)ccc2oc(O)nc2c1 CC1(C)CN(C(c2ccn(C(F)(F)F)n2)=O)CCC1NC(=O)Cc1ccno1 C12(C(=O)NCC(C3CC3)NC(C3CC34CCOC4)=O)CCCCC1NC(=O)CC2 c1(CNC2CCC(=O)NC2c2ccccc2)nc2cccc(Cl)c2[nH]1 c1(C(N2C(C3CCN(C(C)=O)C3)CCCC2)=O)ccc(NS(=O)(=O)CC)cc1C c1(OC)ccc(C)c(NC(=O)CCCNC(C2CCOC(C)C2)=O)c1 CC(C)C(O)CC(=O)N1CCCC1CNC(=O)C=CCF c1(OC)ccc2[nH]c(=NCCCOCCNC(C3CSCC(=O)N3)=O)sc2c1 CCC(O)C(C)(C)C(=O)NOC(CC(C)C)C(=O)N1CCSCC1C C1(CNC(CN(CCC)C)=O)CC(F)CN1C(=O)Cn1nnnc1-c1ccsc1 C1(CC)CN(C(=O)C(F)(F)c2ccnn2C)CCC1NC(c1cccc(O)n1)=O c1(NC(=O)C(Cl)Cl)cccc(CO)c1F CCCCCC(C(=O)N(C1CCCN(C(=O)C(C#N)CC)C1)CC)C(C)C N1(C(C2C3CN(C(COCC=C)=O)C2C3)=O)CCC(C2(C)CC2)C1 C1(NC(=O)C=CC2CCOCC2)CCN(C(c2n[nH]cc2F)=O)CC1F O=C1NC(=O)c2ccccc2C1=CNC1CC(Cc2ccc(Br)cc2)C1 C(=O)(C1=C(Cl)CCOC1)NC1C(NC(c2cc(CCC)on2)=O)COC1 CC1(C)COCCC1C(=O)Oc1ccc(OCc2ccccc2)cc1 C1(NC(c2c(C)nc(CC)s2)=O)CC1C1CCCN(C(C23CCC(C2)OC3)=O)C1 Cc1ccc(COc2ccc(F)cc2)nc1.N1(C)CC(CNC(C2CC2)=O)C1 C(=O)(C(CNCC1(O)CCSCC1)CC1CCCC1)NCCN(CC(C)C)CC C1(NC(C=CC)=O)CCCCN(C(=O)CCSc2ccc([N+](=O)[O-])cc2)CC1 N(C(=NCCF)NC(C)CC(F)(F)F)CC1C(OCC)C1 c1(CN2C(C(=O)Nc3ccc(C)c(C)n3)CC3CC32)ccc(Cl)c(Cl)c1F C1(C(=O)NC(CSCC)C(=O)N(C)CCc2cccs2)CCC(=O)N(C)C1 C(C)(C(C(C)C)NC(=O)CSCc1ncc[nH]1)NC(c1cc(C(C)C)no1)=O C1(C(C)NC(=O)CNC(c2ccoc2)=O)CCCN1C(c1ccccn1)=O C1(C2CCCCO2)(C(=O)NCCNC(=O)C(c2ccccc2F)O)CCOCC1 C1(NC(C2(C(C)C)CCC2)=O)CCN(C(=O)CCCc2n[nH]c(=N)s2)CC1C CC1CC(C(=O)NCCNC(=O)COC2CCOCC2)CS1 c1(C(=O)NC2(CC=C)CN(C(C3CCC(C)C3)=O)C2)cc(Br)c2[nH]nnc2c1 C1(CNC(C2C(CCC)CCC2)=O)CN(C(=O)CNc2ccccc2)CCCO1 N1(C(c2c(OC)nccc2)=O)CC(CNC(=O)Cc2nccs2)CC1(C)C N1(C(CNC(=O)NC2C(C)C2)=O)CCCCC(CC(N2CC(O)(C(N)=O)C2)=O)C1 c1(C(=O)NCCC(CNC(C2(CC)CC2(F)F)=O)O)cnn(C)c1C1CC1 c1(C(N(CCNC(C(C)OCCC=C)=O)C)=O)c(C)nn2c1CCCC2C C1(C(=O)OC)CC2CCC1N2C(=O)CC1N(C(C2CCC(O)C2)=O)CCC1(C)C Cc1cc(C2(NC(=O)C(Cn3cncn3)NC(C3CC(C)SC3)=O)CC2)no1 N1(C(CCCC#CC)=O)CCCC2(CCC(NC(=O)CCCSC)C2)C1 C(C(C)(C)CN(C)C)(c1nnnn1CCCF)NCCCC=CC N1(C(C2(CC=C)CC2)=O)CCCC(COC)(NC(c2ccnn2C(C)C)=O)C1 N1(C(CCN(CC)CC)=O)CCN(C(c2cc[nH]c2)=O)CC1C1CCC1 O=C1CCC2CN(C(=O)NC(c3cccc(OC(F)F)c3)C(F)(F)F)CC2N1 C1(NC(=O)Nc2ccccn2)CN(Cc2cnc(Cl)nc2Cl)CC1(F)F N(C1CCc2cc(Cl)ccc21)C(=O)NC(c1ccc(Br)cc1)CC N(S(=O)(=O)N1CC(C#N)C1)CCCC(=O)OC(C)(C)C N1(C(C2CC(CC)C2)=O)CCC(Cn2cc(CCC3CCCO3)nn2)C1 CC(C)(CCS(C)(=O)=O)C(=O)N1CCCN(C(=O)CC2CCOC2=O)CC1 C1(CCC(=O)N(CCNC(c2ccc(C3CC3)cc2)=O)C2CC2)NC(=O)NC1=O O=C(C#CC1CC(F)(F)C1)NCC1CCCCC1NC(C12CCC(F)(CC1)C2)=O C1(CNC(C(C)=C2CC2)=O)CC2CCC(C1)N2C(C1CCCCCC1)=O N1(C(c2c(CC)cco2)=O)CCOC2(CCN(C(C3COCCOC3)=O)C2)C1 C1(CC(N)=O)CCCN(C(=O)C(C2CCC2)NC(c2cnncc2O)=O)C1 C(=O)(C(F)CCC(C)C)NCC1CCCN(C(c2cncc(C#C)c2)=O)C1 N1(C(COCCCCC)=O)CCCCC1C(=O)Nc1[nH]ccc1CC C1(C(=O)NCC2C(CNC(c3cc(C(C)(C)C)on3)=O)C2)C2(CC2)C12CC2 C(=O)(C(C(C)C)c1ccn(C)n1)NCC1CC(O)(CNC(c2c(CC)csc2)=O)C1 N1(C(CC=C)=O)CCCCC1C(=O)NCCOCC(C)(C)O Cc1cc(F)cc(C(=O)NC23CCCN(C(=O)CN(C)CCO)CC2C3)c1N Cc1cc(F)c(C(=O)NCC2(CCNC(C3C4CS(=O)(=O)CC34)=O)CC2)cc1F CCCC(C(=O)NC1CCCC(NC(=O)Cc2cn(C)nc2Cl)C1)NC(N)=O C1(C(=O)NC2C3CN(C(c4c[nH]c(=N)o4)=O)C2C3)CC2(C1)CC(F)C2 N1(C(CCC=CC)=O)CCN(C(=O)C(COc2ccccc2)OC)CCC1C C=C=CCCC(=O)NCCn1cc(C(=O)NCc2nc(C)cs2)cn1 c1(CCNC(C(Cc2cc[nH]n2)NC(C=C(C)C(C)C)=O)=O)ncccc1F O=C(C1=Cc2ccccc2C1)NCC1(C(N)=O)CN(C(C2C3CC4C(C3)C24)=O)C1 N1(C(c2c(C)n(C)cn2)=O)CC2CC(C1)N(C(=O)Cn1ncccc1=O)C2 CC1CC(C(=O)NCC(=O)NC2CC2)CN1C.C12(CCC1)C(=O)NC2 Cc1cnc2c(C(=O)NC3CCCC34CCN(C(C3(F)CC3)=O)C4)cnn2c1 C12(NC(c3cccc(C)c3F)=O)CCN(C(c3nn(C)cc3N)=O)CCC1C2 N1(CC)CC(C(N2CCCCC2CNC(=O)CS(=O)(=O)N(C)C)=O)CC1=O Cc1cc(C(=O)NC23CC(CNC(=O)C(C(C)C)N(C)C)(C2)C3)ncc1F CCC(CC)(CN=c1[nH]cnc2cc(Br)ccc12)NC(C1CC=CCO1)=O C1(NC(CN2C(C)CC2)=O)CCN(C(=O)C2=CCCSC2)CC(C)(C)C1 c1(C(C)C)cccc(C(=O)NCC(C)NC(=O)C(O)CN2CCOCC2)c1 C(=O)(C1Cc2ccccc21)N1C(C)CCC(NC(C2CCS(=O)CC2)=O)C1 C1(CNC(C=C(COC)C)=O)CCC2(CC1)CCN(C(c1nn[nH]c1Cl)=O)CC2 c1(Cc2ccc(OCc3n(CC)c(C)nc3)cc2)ncnc2cnccc12 c1(C(=O)NCC2CN(C(CNS(CC)(=O)=O)=O)CC2C)cncc(C)c1C c1(C(=O)NC2(CNC(CCCc3scc(C)n3)=O)CC2)ccc2c(n1)OCCO2 C1(C(N2CC(CCNC(c3cc(CC)no3)=O)C2)=O)CC2CCCC(C1)C2(F)F CCC(O)C(C)(C)C(=O)N(CCNC(=O)C(c1ccccc1)SC)CC C(=O)(C(F)C(=O)NCCOCCN(C(c1conc1CC)=O)CC)OCC Cc1cc(F)ccc1C(=O)NCC1CN(C)CCN1C(=O)CCCc1cnn[nH]1 NS(=O)(=O)C1CC(C(=O)NC2CC(NC(c3cc(C(F)F)ccc3Cl)=O)C2)C1 C12(CNC(=O)Cc3cnns3)CCC(C(=O)NCC3C=CCC3)(CC1)CO2 C1(NC(c2n(CC=C)ccn2)=O)(CO)CCCN(C(c2ccc(C)s2)=O)C1 C1(CCC)CN(C(c2cnc(C3CCC3)s2)=O)CCN1C(=O)C(O)C1CC1.CCO N1(C(C2(C#N)C(C)(C)C2)=O)CCCC(C(=O)NCC2CSC2)(CO)C1 C1(NC(C2(NC(C(C)=C3CCC3)=O)CC(F)C2)=O)CCOCC1F CC1(C)CCCC1CCNC(=O)NCCC1(c2ccccc2)CCCO1 N1(C(c2cc(C)[nH]c2)=O)CCCC(C2CN(Cc3ccc(C(C)(C)C)cc3)C2)C1 c1(C(=O)NCC(C#C)OC)[nH]ccc1CNC(=O)C(C)C N1(C(Cc2c(C)non2)=O)CCC(O)(CNC(=O)COCc2cccnc2)CC1 c1(CNC(C(OC)OC)=O)cc(C(=O)NC(CN2CCCC2)CO)co1 c1(C(=O)NC2C(NC(C(=O)NCC)=O)CCCC2)nn(C)c2c1CSCC2 CC(C(=O)NCC1CN(C(=O)C=Cc2ccncn2)C1)C(C)S(C)(=O)=O c1(C(=O)NCC2C=CCN2C(=O)Cc2nc[nH]n2)ccc2nsnc2c1 N1(C(c2c(C)nsc2C)=O)CCCCC2(C1)CN(C(C1(C3CC3)CC1)=O)C2 c1(NC)ccc(C(N2CC(OC)C(NC(=O)CCn3c(O)nnc3O)C2)=O)nc1 c1(C(=O)NCC(CCNC(CC(CC)C)=O)O)cccc(C)c1N N1(C(c2cccc(SC)c2)=O)CCC12CCN(C(c1cc[nH]n1)=O)CC2 C1(O)(C(C)NC(c2nnc(C)s2)=O)CCN(C(=O)CCCc2cccs2)C1 C1(C)(CNC(CCC2(C)CC2)=O)CCN(C(=O)Cc2ccco2)CC1 c1(CC(=O)NC2CC(O)(CNC(C(C)OC)=O)C2)ccccc1C(F)(F)F N1(C(CC(CN(C)C)O)=O)CCC(C)(C)C(CNC(=O)CCSCC(N)=O)C1 N1CCOC(SCC)C1.c1(CC(=O)N)cc(C2CC2)no1 C(=O)(C(C)(C)CCC#N)NCC(Cn1cc(CNC(C(C)O)=O)nn1)(C)C C1(NC(=O)NCCCOCCOC)CCOC2CC12 Cc1cnc(C(N2CC(CNC(c3cccc(C(F)F)c3)=O)C2)=O)c(F)c1 Cc1ccncc1CN(C)C(C1CC(NC(=O)CCCCC2CC2)C1(C)C)=O C1(NC(CC(C)C)=O)CCN(C(=O)C(C(C)C)n2ccnc2)CC1 CC1(C)COC(C(=O)NC2COCC2C(=O)NCC2CCC(C)(C)O2)C1 n1(CCC)nccc1C(c1nnnn1-c1ccccc1)NCCCn1ccnc1 Cc1[nH]nc2c(C(=O)NC(C)(CNC(c3ncccc3Br)=O)CO)cccc12 Cc1nc(C(C)C)ncc1C(=O)NC(CNC(=O)CN1CC(C)C1)C(C)C(C)C CCC(CC(F)(F)F)C(=O)NC1(CNC(=O)C(C(=O)OCC)SC)CC1.C(C)(C)C C1(=CC(N2CCC(CCCCNC(C(C)O)=O)CC2)=O)CCC(C)(C)CC1 C1(CC(=O)NCc2cccc(C#C)c2)CCC(C)(C)N(C(=O)C=CCCC(C)C)C1 c1(CC)ncc(CN2CC(=O)N(CC(c3cccnc3)N(C)C)C2)cn1 c1(CC)ccnc(C(N2CCC(CN(C)C(C3(C4CCCO4)CC3)=O)C2)=O)c1 C1(C(=O)NC2C(C(=O)NCC3OCCN(CC)C3)CC2)CC(C)(C)CCO1 c1(C(=O)NC2(CC(=O)N(CC=C)C)CCC2)cc(O)nc(O)n1 Cc1ncccc1CC(=O)N(CCC(=O)NCC1CC1C)C c1(C(N2CCCC(CNC(C(CCC)NC(N)=O)=O)C2)=O)ncc2ccccn12 c1(C(=O)NC2CC(C)N(C(C)C)CC2)cncc2ccccc12.c1ccc(Cl)[nH]1 N1(C(CCC(=O)NCC)=O)CCC(CNC(C2(Cl)CC2(C)C)=O)C(C)C1 c1(C(=O)NC(CNC(C2(CC)CCNC2=O)=O)C(C)(C)C)nc2c(s1)CCCC2 c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CC2)ccc(O)c(Cl)n1 C(C1=NOC2CN(C(=O)CCCS(N)(=O)=O)CC12)NC(c1noc(CC)c1C)=O C1(C(=O)NCC2C(C)CN(C(=O)CC3(O)CCOCC3)C2)CC2(CCCC2)CO1 C1(C(=O)O)CCC(COCc2ccccc2)N1C(C1CCCC(=O)O1)=O N1(C(C2CCC(C)N2C(=O)CNC(=O)C2CC2)=O)CCNC(=O)CC1 c1(C(N(C)CC2CCN(C(CCOCC(C)C)=O)CC2)=O)cc(C#N)ccc1N c1(OC)ccc(Cl)c(F)c1C(N1C2CCC1CN(C(C1C3CCCC13)=O)C2)=O n1(CC(N2CC(CC(C)NC(C3C(C=C)C3)=O)C2)=O)c(=O)oc2ccccc12 C#Cc1cnc(C(=O)NCCN(C(=O)C(C(C)C)C(C)C)CC)c(C)c1 N1(C(C=C2CCC(C)C2)=O)CCCCC2(CCN(C(=O)Cn3cccc3)C2)C1 C1(NC(CCSCCCC)=O)CN(C(=O)Cc2cnns2)C(C)(COC)C1 C(=O)(C1=NOC(C2(O)COC2)C1)N(C(CNC(c1cc(C)ncc1)=O)C1CC1)C N1(C(c2nc(C(C)(C)C)oc2)=O)CC2CC1C2CNC(=O)CC1(O)CCOC1 Cc1cc(C)c(CSCC(N2CC(c3cc(O)no3)C2)=O)s1 CC1(C)C(CN2CCN(Cc3ccccc3)C(=O)C2)C(C)(C)C1O c1(CCNC(C(C2(C)CC2)NC(C2C(CC)OCC2)=O)=O)cnn(C)c1C C1(C)(C(=O)NCCCN(C(c2n(CC)ncc2)=O)C(C)C)CCCCC1 N1(C(Cn2c(C)ccn2)=O)CCC(C(C)NC(c2cc(CO)on2)=O)CC1 c1(C(=O)NC(CNC(C2(CF)CC2(F)F)=O)C2CC2)csc(CO)n1.C1CC1 CCC(O)C(C)(C)C(=O)NCCN(C(=O)Cc1ccnn1C)C Cc1cc(C(=O)NC2CN(C(=O)C=CS(C)=O)C2)c(F)cc1F C1(C(=O)NCC2(O)CN(C(c3c(CC)ncs3)=O)C2)CCN2CCOCC12 C(=O)(C(F)(F)C(F)(F)F)NCC(CNC(c1cccc(CC(=O)OC)c1)=O)O c1(C(N2C3C(N(C(COCC(C)C)=O)C)CC(C3)C2)=O)ccc2oc(=N)[nH]c2c1 c1(N2CCN(C)C(CO)C2)nc(N2CCCC(CF)C2)nc2ccc(Cl)cc12 c1(CC)onc(C)c1C(=O)NC(C)CC(C)NC(C1(CC)CC(C)(C)C1)=O C1(CNC(c2cncc(C)c2)=O)CN(C(C2CCC2)=O)C2(CCOCC2)C1 C(C(CNC(c1ccc(C(F)F)cn1)=O)C(F)(F)F)NC(C1OCCC(C)C1)=O C1(OCC(=O)NCCC(=O)NC(COC)(C)C2CC2)CC(F)(F)C1.C1(OC)CCC1 C1(C(C)(C)C)CCN(C(=O)C2=NOCC2)C(CNC(C2(C3CC3)CC2)=O)C1 C=CCCCCCC(=O)N1CC(CNC(=O)CCCn2nc(C)nc2C)CC1C N1(C(CC(CNC(c2cnc(C)s2)=O)O)=O)CCC2C(C(N)=O)C2C1 C(=O)(C(C)(F)C(=O)NCC(C1CCN(C(C2CCOC2)=O)CC1)(C)C)OCC C(C)(CO)(C(=O)N1CCCC(C(C)NC(=O)CCCOC(C)C)C1)OC n1(CC)nnc(C(=O)N(O)Cc2cn(CC(=O)C(C)(C)C)nn2)c1C Cc1ccc(C(=O)NCC(C(=O)NC2CC3(CCCO3)C2)C(C)C)c(C)c1 c1(C(=O)NC2C=CCN(C(c3c(C)occ3)=O)C2)ccc2ccnc(O)c2n1 C(C(C)(C(=O)NC)OC(CCO)C(F)F)N.c1(OCC(=O)NCCOC)ccn(C)n1 C1(CC(N)=O)(NC(C(C)OCC#C)=O)CCN(C(C2CCCC(C)(C)C2)=O)CC1 Cc1cc2[nH]c(C(=O)NCCCCCc3cn[nH]c3)cc2o1 Cc1cccc(C)c1CC(=O)NCCCCCN(C(=O)Cc1cncc(F)c1)C c1(Nc2cc(C)sc2-c2ccccc2)cccc(Br)c1CO.C12CC1NC(=O)N2 c1(NC(CCNC(c2c(C)c[nH]n2)=O)=O)cccc2ccncc12 c1(C(=O)NCC2C(CNC(c3cncs3)=O)C2)c[nH]c2ccc(Cl)cc2c1=O Cc1cc(N(C)C(C2CN(C(c3coc(C(N)=O)c3)=O)CCO2)=O)cc(F)c1 N1(C(CCOC(C)C)=O)CCC(O)(CNC(C2C3CCC2(c2ccco2)C3)=O)C1 C1(C#CC(=O)N(CC(C)CNC(=O)CC2(C)CCCC2)C)(CC)COC1 CC1OC2(C(=O)NC3CCCN(C(c4ccc(=N)[nH]n4)=O)C3)CC1C2 N1(C(C2C(c3cccc(OC)c3)C2)=O)CCC2(CCCN2C(=O)CCCCCl)C1 C1(C(=O)NC(CCNC(CC2N(CC)CCOC2)=O)(C)C)CCCCCC1(F)F Cc1ccc(CC(=O)NC(CC(=O)NCCC2CCC2)C2CC2)cn1 C#CCC(C(=O)N1CC(C)(O)C1)NC(=O)CC1CCCCCC1 C(=O)(CCCC(=O)NC(C)C(C)NC(=O)C(C)(C)C1CCOC1)NCCC C1(C(N2CCC(C)(CCC)C2)=O)CCCCN(C(c2snnc2C)=O)C1 Cc1cc(C#N)ccc1-c1nc(C(=O)NCCc2cnc[nH]2)cs1 N1(C(c2ccn(C)c2)=O)CC2CC(NC(=O)Cn3ccc(C(F)F)n3)C2C1 c1(C(N2CC=CC23CCCC3)=O)c[nH]c2cc(Cl)ccc12 Cc1c(F)ccc(N)c1C(=O)NCC(C)CNC(C1CCCN(CC(F)F)C1)=O c1(C(=O)NC(C)CNC(C2CC(C(F)F)C2)=O)csc(C2CC2)n1 C1(NC(c2cc(C)cc(O)n2)=O)CC2CC1CN(C(c1cc3occc3s1)=O)C2 Cc1cc(=NC2CC(CN(C)C)C2)[nH]c(N2CCC(C)(c3cccc(F)c3)C2)n1 CCCC(CCCO)C(=O)NC1(C)CN(C(=O)C(C(C)C)c2cnn(C)c2)C1 c1(C(=O)NCCNC(CCCCCC=C)=O)noc2c1CC(C)CC2 CC1(C(=O)NCC2CC2NC(c2cnoc2-c2ccc(Cl)s2)=O)CC(F)C1 N1(C(CC(C)=C(C)C)=O)CCCCC(CNC(c2cnc(C3CC3)[nH]2)=O)C1 c1(C(=O)NC(c2cnc(-n3c(C)ncc3)nc2)C)ccc(Cl)c(Cl)c1 Cc1cc(C)n2cnc(C(N3CCC(NC(C4(C)CCCOC4)=O)CC3)=O)c2n1 N1(C(c2cc(C)on2)=O)CCC(C(=O)NCCOCC(F)(F)F)C12CC2 c1(CC)ccc(C=CC(=O)NC(C)CCNC(=O)Cc2ccc(C#N)cc2)cc1 c1(CC)[nH]nc(C(=O)NC2C3CCN(C(c4cccnc4)=O)CCC23)c1[N+](=O)[O-] c1(CCC)nc(NC(=O)NCCCC2(O)CCC2)cs1 c1(C(=O)NC2(C(=O)Nc3cn(CC=C)nc3)CC(F)C2)ccc(O)cc1 N1(C(CC(C)(C)C)=O)CCOC2(CCCN(C(=O)CC3CCC(=O)NC3=O)C2)C1 c1(C(CC)=O)cc(C(F)(F)F)ccc1C(C)C.C1(CNC)CCCN(C(=O)CON)C1 C1(C(=O)NC2(C)CCN(C(CC(CC)O)=O)CC2)CCCCC1C1CC1 N#Cc1cccc(OCC(=O)Nc2ccc(-c3cn(CCF)nn3)cc2)c1 c1(CC(C(=O)N(CC(CC)NC(c2cc(OC)ns2)=O)C)O)ccc(OC)cc1 C(CC(C)CC)(C(=O)N1CC(C2=NOCC2)C1)NC(C(=O)NCC)=O c1(C(N2CC(C(N)=O)(CNC(c3n(C)nnc3)=O)C2)=O)cc(F)cc(Cl)c1O O=C(CC(C(F)F)n1ccnc1)NCc1cn(CCNC(C2C3CCC23)=O)nn1 C#CCC(CC(=O)NCCOC)NC(C1CCCC(=O)CC1)=O C(=O)(N1OC2C=CC1CC2)C1N(C(C(C(C)C)(C)C)=O)CC(=O)C1 Cn1c(C(=O)NCC2COCCN2C(=O)CP(C)(C)=O)cnc1Cl CC(CC(C)(F)F)C(=O)N(CCNC(=O)C(F)(F)Cc1ccccc1)C1CC1 CS(=O)(=O)C=CC(=O)N1CCOCC(NC(c2c(F)cncc2Cl)=O)C1 CC(=O)C(C)(C)CC(=O)N(C(C)C(N1CCCC1(CO)CO)=O)C C12(CNC(CCc3cncc(C)c3)=O)CC(NC(=O)CC3=CCCC3)(C1)C(C)O2 C1(C)(CN(C(c2c(C)nn(C(C)(C)C)c2)=O)C)CCCCO1.c12cn(nn1)C2 C(=O)(C(CC)C(C)O)NC(CNC(c1n(CCC)ncc1)=O)C CCCCCC(C)(C)C(=O)Nc1cc(F)c(Cl)cc1Br N1(C(c2c(C)ncc(Cl)c2)=O)CC2CCCC2(NC(=O)C=C2CCC(C)C2)C1 CC1COCCC1N(C(=O)C(F)CC1CN(C(c2ccncc2N)=O)C1)C CCCC(C(N)=O)NC(=O)C(CCC1CC1)NC(=O)CN(C)C(C)=O NS(=O)(=O)c1cccc2c1CCN(N1CCCC1C1CCCCC1O)C2 N12CCCCC(C1)N(C(=O)C(C)CC1CCC1)CC2=O.c1(CCC=CC)ccccc1 c1(C(=O)NC2C(CNC(c3cnc(C)[nH]3)=O)C2)cncc(C(F)(F)F)n1 n1(C(C)C)cc(CC(=O)N(CC(C2CC2)NC(=O)CSCCN(C)C)C)cn1 N1(C(c2conc2C2CC2)=O)CC(NCc2nc(CC)on2)CCC1C C(C(=O)NCCCOC)(C1CCCC1)OCCC=C.C1(C2(C)CC2)C(=O)N1 N1(C(=O)NNc2ccccc2)CCCC1C1CCCN1c1ccncc1 c1(C(N2CC3C(CNC(CCOC)=O)(C3)C2)=O)cc(F)ccc1I c1(C(=O)NC(C2CCN(C(Cn3ccc(C)n3)=O)C2)C)cc2c(F)cccc2[nH]1 c1(C(N2CC=C(CNC(C3C=CCCC3)=O)CC2)=O)n[nH]c2c1CSCC2 C1(n2cc(CCCC)nn2)CCC(C=O)CC1.CN1CCCC1C1(C(=O)OC)CC1 c1(C2(CN(CCC#C)CC)CC2)ccncc1 N1(C(c2c(C)cc(O)nn2)=O)CCC2CCCC12CNC(=O)CCS(C)(=O)=O N1(C(CCCc2n[nH]c(=N)s2)=O)CCCC(F)(CNC(C2CC(Cl)(Cl)C2)=O)C1 CCC(CC(=O)N1CC2CC1CN(C(=O)C(C)SC)C2)C(C)C CC(CC(F)(F)F)C(=O)NCC1(C)CCCN(C(c2ccc(N=[N+]=[N-])cc2)=O)C1 c1(C(N2C(CNC(C(CC=C)NC(C)=O)=O)C=CC2)=O)nc(OC)ccc1C CCC(CC(=O)NC1CC(NC(c2c(C)nsc2C)=O)C12CCC2)C(C)C CCCCC(C)C(=O)N1CCN(C(=O)CCOc2ccc(CC)cc2)C2CC12 C(N=c1[nH]c2cc(F)c(F)cc2[nH]1)c1c(COC)nn[nH]1 C1(C(C)(C)C)CCN(C(c2cnc[nH]2)=O)C(CNC(C2CC2c2cc[nH]n2)=O)C1 N1(C(c2c(CC)nc(C)s2)=O)CCN(C)C(CNC(=O)C(F)C2CCC2)C1 C(C(=O)NC1(CO)CCN(C(=O)Cn2cc(C3CC3)nn2)C1)(C(C)C)SCC C12(Oc3ccc(OCC)cc3)CCC(C1)C(C)(C)O2.C1C(=O)N1.C(=O)(CSC)N(C)CC C#CC1(O)CN(C(C2CSCN2C(c2sccc2CO)=O)=O)C1 C1(C(=O)OC(C)(C)C)CC2(C1)CC(CS(=O)(=O)NC(N)=O)C2 N#Cc1c(Br)cccc1S(=O)(=O)Nc1cccc2c1ccn2CCO C1(C(N(C)CC2CCCOC2)=O)(NC(C2CCCN2C2CC2)=O)CCSC1 C#CCCC(O)C(=O)N1CCC(CNC(c2ccncc2Br)=O)(OC)C1 C#CC1(C(=O)NC(C)C=CC(=O)NCc2cnc(CC)[nH]2)CCCC1 c1(CCC(N2CC(F)(CNC(=O)COC3CCCC3)C2)=O)cccc(O)c1 n1(CC)nc(C)cc1-c1nc(-c2cccc(C(F)F)c2)nn1CC1CCCO1 N1(C(C(C)=C2CC2)=O)CC(C)CC1C(=O)NCC(C)(C)C#N c1(C(=O)NCC2(CCNC(CSC(C)C)=O)CC2)cnn2c1SCC2 C(=O)(C1=CS(=O)(=O)c2ccccc21)NCC1C(NC(CCNC(=O)C=CCl)=O)C1 C(=O)(C(CNC(C1CC(C2CC2)=NO1)=O)C(C)C)NC1C(CC)CCCC1 N1(C(=O)CCOc2cccc(Cl)c2)CCN(C(=O)CC2CC2)C(CC(F)(F)F)C1 C1(C(=O)Nc2cccc(Cl)n2)CC12CCN(C(=O)C=Cc1ccoc1)C2 CN1CC(C(N2CCN(C3CN(C(C4COC(=O)N4C)=O)C3)CC2)=O)NC1=O c1(CCC(=O)NC2C(NC(C(C=C)c3ccccc3)=O)COC2)ccnc(C)n1 Cc1ccn(C)c1C(=O)NCCc1cc(C(=O)NC2CCS(=O)(=O)C2)no1 S(=O)(=O)(c1cccc(=NCc2ccco2)[nH]1)NCc1scc(C(N)=O)n1 C=CC1(CC(N2CCC(COCC)CC2)=O)CN(C(=O)CC2CC2)C1 Cc1ccc2c(C(N3CCC(NC(C4CCC4(C)C)=O)C3)=O)ccc(O)c2c1 C1(CNC(c2ccc(OC(F)F)cc2)=O)CCCCCN1C(=O)C=C1CCC1 C(C)(N=c1nc2scnc2c(NCc2ccc(Cl)c(Cl)c2C)[nH]1)c1scc(C)n1 N1(C(C2CN(C)C2)=O)CC2(C=C(C(=O)N3CCCCCC3)CO2)C1 N1(C(C(C)SCCCC)=O)CCC2CC2(C(N2CC(OCC(N)=O)C2)=O)CC1 C(=O)(CC1=CCN(C)CC1)N(C1CCC12CCNCC2)c1ccnc(C)n1 C(=O)(CCCC(N)=O)N(C1CCN(C(C(CC)C)=O)C1)C C(=O)(CS(=O)(=O)C1CC1)NCC1(CNC(C(C2CCCOC2)OC)=O)CCC1 CCC(CC)CCC(=O)N1C(C)C2CC1C2NC(=O)Cn1ccnc1C(C)C C12(CNC(CC(C)OC)=O)CCCC(CN1C(c1ccccc1C(F)(F)F)=O)C2 C1(CNC(C2ON=C(C(C)C)C2)=O)(NC(=O)C=CCO)CC2CCC1CC2 N1(C(CC)C(C)C)CCc2ccc(Cl)c(F)c2C1C C(=O)(CCCC(F)(F)CO)N1CCC(CCNC(c2c(C)cc(C)[nH]2)=O)C1 c1(C(N(CC(CN(C(=O)COCCF)C)O)C)=O)cc2n(c1)CCC2 C(=O)(C1CCc2ccccc21)N1CC2CC(NC(c3c(Cl)ncc(C)c3)=O)C2C1 C(c1ccc(Br)o1)=CC(=O)CNC1CC=CCC1 C(=O)(CCCNC(N)=O)N(CCN(C(C(C)OC)=O)C)C CCCCC(O)C(=O)N1CCOC(CCNC(=O)CN(c2ccc(Cl)cc2)C)C1 C1(NC(c2cn(C)c(=O)n2C)=O)CCCCC12CCN(c1cncc(Cl)n1)CC2 N1(C(C(N2CCOCC2)C)=O)CCOCC1CC(=O)Nc1cccc(CO)c1 CC(C(=O)N(CCCOCC1(CSC2CCC2)CC1)C1CCC1)N(C)C S(=O)(=O)(c1nc(NC(C=C)C2CC2)ccc1Br)N(C1(C2CCCCC2)CC1)C C1(C2(O)CCN(C(C3CCN3S(C)(=O)=O)=O)CC2)(NC(C=CCCC)=O)CC1 c1(C(N2CCN(C(N3CCN(C(N(C)C)=O)CC3)=O)CC2)=O)cc(Cl)ccc1I CCCCC(CC)C(=O)N(C1(CNC(=O)CC2(C(F)F)CC2)CC1)C N1(C(C(CSC)C)=O)CCC(CNC(C2CCCN2C)=O)C(F)(F)CC1 C1(C(=O)NC(COC)COC)CC(O)CN1C(c1cn(C)nn1)=O N1(C(CC2(C)CCCO2)=O)CC(S(=O)(=O)NCc2ccccc2)C1 CC1CC(C(=O)NCC(=C2CN(C(=O)CCN3CCCCC3)C2)F)CC(C)C1 CCCC(C#N)C(=O)N1CC(O)CC1CNC(=O)C(C1CC1)OCC N1(C(C(C(C)O)N(C)C)=O)CCCCCC1C(=O)NCC(n1cccn1)C c1(C(C)C)ccc(C(=O)COC(=O)C(c2cnn(C)c2)C)cc1 C1(C(N2CCN(CCNC(c3n(C=C)ncc3)=O)CC2)=O)CC2C(C1)C2(F)F N1(C(CC2(CSC)CC2)=O)CCCC(CO)(NC(C2CCS(=O)(=O)N2)=O)C1 c1(C(=O)NCC2N(C(c3c(CCC)ocn3)=O)CC2)cc(CC)c(=O)n(C)c1 C1(COC)(NC(=O)Cc2ccsc2)CCN(C(C2(C)CC2(C)C)=O)C1 C(CN=C(NCCN1CCCCC1)NCC1CC1(C)C)c1cc(C)no1 S(=O)(=O)(c1cc2sc(=NC(C)c3nccs3)[nH]c2cc1Cl)NC1CN(C)C1 N1(C(c2c(C)occ2)=O)CCC(C2CC(NC(=O)Cc3cc(F)ccc3F)C2)C1 c1(CN(C(CCCC=C)c2ccccc2)C)nc(C)c(C)n1CC c1(C(=O)NCC2N(C(C=CC)=O)CC=C2)ccc(C)c(CO)c1 CC(C)CC(C(=O)NCc1cnco1)NC(=O)CCC1CC1C N1(C(c2c(C)nc(C)s2)=O)CCC2C1CCN2C(c1ccc(F)c(Cl)c1F)=O C(C(C)C(C)C(=O)NCC(C)(C(C)C)NC(=O)COCc1ccncc1)OC CCCCC(CC)CC(=O)NCC1CCN(C(=O)C(C)SC(C)C)C12CCC2 Cc1cccc(C)c1C(=O)NC(C1CCN(C(c2csc(C)c2C)=O)C1)C c1(C(=O)NCC2C(NC(CC3N(C)CCOC3)=O)C2)cc(S(N)(=O)=O)ccc1Cl CC1=C(C)CN(c2nnc(-c3ccc(-c4cccc(C(C)C)c4)cc3)n2C)CC1 C1(CC)CCCN(C(=O)CC2CCN(C(C3(CO)CCCCC3)=O)C2)CC1 c1(C(=O)NC2CC(NC(CCC(C)OCC)=O)C2)cc([N+](=O)[O-])ccc1CC c1(COCCCNC(c2ccc(C(=O)NC(C)C)cc2)=O)cc2c(s1)CCC2 C(c1ccccc1)=CCC(=O)NCC(C(=O)NC(c1cccs1)CC)C Cc1cccc(C(F)C(=O)NCC2(CNC(C3CCSC3)=O)CC(F)(F)C2)c1 CCC(CN(C)C)CC(=O)NC1C2CC1N(C(=O)CNC(=O)C1CC1)C2 c1(SC)ccc(C(C)Sc2cn(CCCF)nn2)c(O)c1Cl C1(C(C)C)CCN(c2cc(-c3ccccc3)nn2C)C(=O)N1.C=C1CC(C)C1 C(=O)(C(F)CC(C)(C)NC(=O)C(O)CN(C)C)NCc1ncc(CC)o1 c1(OC)cccnc1C(F)(F)C(=O)N(C(F)CO)CCO c1(C(C)NC(c2n(CC(=C)C)nnn2)c2occc2CC)ccc2c(c1)CCC2 C(C(=O)NNC(=O)Nc1cnc(NC(=O)CCCC(=O)CC2CC2)s1)SCCOC c1(C(=O)NC2CCCCN(C(COCCOCC)=O)C2)cc(C)c(Cl)cc1F N1(C(Cc2ncn(C)c2)=O)CC2CCN(C(=O)COCCF)C2C1 C#CCCC(C(=O)NCC1(CO)CC(C)C1)NC(=O)CCC(C)CC C1(C2(C=C)CCC2)(C(N2CC(C=C)C(NC(=O)C(C3CC3)SC)C2)=O)CCC1 c1(O)cccc(C(C)=O)c1.CCC(C)C(=O)NCc1ccoc1C(=O)NCC C1(C(=O)NC(CNC(C(C)SCC)=O)(CC)CC)CCC2(CCC2)C1 c1(C(=O)NCCN(CC)Cc2ccc(F)cc2F)cc(Cl)cc2cc[nH]c12 N1(CCOC)CCN(C(=NCCc2nccs2)NCc2cnc3n2CCC3)CC1 n1(C2CN(C(=O)OC(C)(C)C)C2)cc(C(=O)OCCCO)nn1.C1CO1 C1(C(=O)NC2(CNC(C(C)OCCC=C)=O)CC2)CCCC(F)(F)C1 CC1CN(C(=O)C=CCN2CCCC2)CCN(C(C2CCCCC2(F)F)=O)C1 C(CCC(CCC)C1CC1)OC1CN(CCCCCCC)C1 N1(C(Cn2cc(C(C)O)nn2)=O)CCN(C(C2CC(O)CN2C)=O)CC2(CC2)C1 C=CC(C)(O)CC(=O)N(CCC(C(C)(C)C)NC(=O)C=Cc1ccc(C)cc1)C C1(NC(C(C)OCC=C)=O)(CNC(=O)C=Cc2cnc[nH]2)CCC(C)(C)CC1 Cc1cc(C(=O)NC2(C)CC(NC(c3coc(CO)c3)=O)C2)n2ncnc2n1 C1(NC(CN(c2ccccc2)C)=O)CCCN(C(C2(C)CCC3CC3C2)=O)CC1 c1(OC)ccccc1CNC(=O)NC1CCC(c2ccccc2)C1 C1(CNC(C(CC)C)=O)CN(C(=O)Cc2ccc(O)cc2Cl)CC1(C)C CC(C)(C)C(C(=O)N1CCCC(NC(=O)C=Cc2cccnc2)CC1)C1CCC1 C1(NC(C(C)N2CCCC2)=O)CCC(CC(=O)NCc2cscn2)CC1 c1(CN2CCC(CNC(c3cccnc3)=O)C2)cccc2cccnc12 C#Cc1ccc(C(=O)NCC23CCN(C2)C3=O)nc1.C1(C(N)=O)(SC)CC1 C1(NC(c2c(N)cc(F)cc2)=O)CC2CCC1C(NC(=O)COC1CCC1)C2 c1(N(CCOCC)CC)nc2ccsc2c(=NCc2cnc(C)[nH]2)[nH]1 C(=O)(C(C)(O)C(F)(F)F)NC1CN(C(c2c(OCCC)cccc2)=O)CC1CC c1(C(=O)NC2CCCC(C(=O)NC3COC(C(F)F)C3)C2)cnn2ccccc12 Cc1cc2ccc1c(=O)[nH]2.C1(OCC(=O)NCC2(NC(N)=O)CC2)CCOC1 C1(CC)C=CCN(C(=O)CC(C)(C)NC(=O)CS(=O)CC)C1 N1(C(c2c(C)ccc(Cl)c2O)=O)CCC2CC1CN(C(=O)COC(C)C)C2 C1(C(=O)NC2(C)CN(C(=O)C3=C(Cl)CCC3)C2)CCN(S(N)(=O)=O)CC1 CC1=CCC(NC(=O)CCC2CCCN2C(=O)C#CC2CC2)CC1 N1(C(=O)NC2CC=CCC2)CCCc2c(F)cc(F)cc21 c1(SCC)ccc(C(=O)N(CCCCN(C(=O)CN2CC3CC3C2)C)C)cc1 Cc1ccc(-c2cc(C(=O)NCCCC(C)NC(c3cncs3)=O)no2)c(C)c1 N1(Cc2c(COC)cccc2)C(=O)NC(c2cnccn2)C1=O N1(C(C(=O)NC(CC#C)CC)=O)CCCC(O)(C(C)C)C1 C12(C(=O)NCC(C)NC(c3c(OC)noc3C)=O)CC3CC(F)(C1)CC(F)(C3)C2 C(=O)(C1=CN=C2N=CNN2C1)N1CCC(CNC(C2CC=CCC2)=O)C1 N1(CC)CCC(CN)CC1.c1(CC(C(=O)CCN(C)C)=O)nccn1C c1(C(=O)NC2(C(N(CC(=O)N(CC)CC)C)=O)CC2)ncnn1C1CC1 C1(C(C(=O)NCC(C)CN(C)C(C2(CO)CC(F)(F)C2)=O)O)CCCCCC1 CCCCC(F)C(=O)NC(CSC1(c2cc[nH]n2)CC1)C(=O)NC c1(NC(=O)NC(CN(CC(=O)NC(CCC)C)C)C)ncc2ccccn12 C1(NC(c2c(C)cc(C)s2)=O)CS(=O)(=O)CC1NC(=O)CN1CC(C)(C)C1 Cc1coc(C2CC2)c1C(N1CC(C)(NC(=O)C(F)OC(F)(F)F)C1)=O CCC(F)(CNC(=O)C(C)(C)C1CCCN1C(=O)CC(=O)OCC)CC C1(C(=O)NCC2CC23CC3)CC2(CCN1C(=O)CCc1ccco1)CC2 C(C1CCN(C(C2CCCCOC2)=O)CC1)=CC(=O)N(C1C(C)C1)C c1(C(N2CCCC(CC(=O)OC(C)(C)C)C2)C(=O)NCC=C)csc2cncn12 C1(N(C)Cc2ccc(C(=O)OC)o2)CCN(C(C2CC(O)C2)=O)CC1(C)C n1(CC(=O)N(C2CCN(C(c3n[nH]cc3Cl)=O)C2)CCC)cc2ncccc2n1 CCC(C)CCCC(=O)NCCN(C(C1OCC2CCCC1C2)=O)CC1CC1 c1(OC)ccc(NC(C2(NC(=O)C(C)N(C(C)=O)C3CC3)CC(O)C2)=O)cc1 C(CCCCCC(=O)N1CCC1C1CCOCC1)NC(CCCC)=O CC(C)C(CO)CCNC(C1COCC1NC(=O)Cc1ccco1)=O CCCCC(C(=O)NC(CC(=O)NCCCCC1CC1C)C(F)(F)F)C(C)C C1(C(=O)NC(CC)CNC(c2c[nH]c(C(N)=O)c2)=O)CC2CC(C1)C(=O)N2 C(=O)(CCCONC(c1cc(OC)cs1)=O)OC.C1(=O)CCCN1C(C)C C(=O)(C1CCCc2nc[nH]c21)NC1CCC(C)N(C(c2cnc(C3CC3)o2)=O)C1 C1(C(=O)NCC2CN(C(C#CC3(C)CC3)=O)C2)Cc2cccc(F)c2O1 c1(CCCNC(C2(C)CN(C(C3CC3C3CC3)=O)C2)=O)cccc(F)c1 N=C(N)NC(Cc1ccccc1)C(=O)N1CCC(c2nc(=N)[nH][nH]2)C1 c1(C(=O)NCC=CCNC(C(CN(C)C)(C)C)=O)c(N)c(F)cc(F)c1F c1(C(N2C(CNC(C(C)O)=O)C=CC2)=O)ccc2ccccc2c1F N1(C(C)=O)CC2CC2(CNC(c2nc(C)oc2-c2ccccc2)=O)C1.C(CCC)(C)=CC N1(C(C2(C)C(C)C2)=O)CCC2(C(=O)NC(c3ccc(O)cc3)CO)CC2C1 C1(OC)CN(C)C(C)(C(=O)NC(CNC(c2nc(Cl)sc2C)=O)C2CC2)C1 c1(OCC)ccc(CC(N2CCC(N(C(=O)CC3(CSC)CC3)C)C2)=O)nc1 c1(C(=O)NCC(CNC(COC(CC)(C)C)=O)OC)cc(Cl)n(C)n1 Cc1ccc2cc1S(=O)(=O)N2.c1(C2N(C(C3CCOC3)=O)CC2)ccc(F)c(F)c1 C1(C(=O)NCCNC(C(CC(C)C)C)=O)Cc2ccccc2C(C)(C)C1 N1(C(c2c(CNC(C3(C)CC(=C)C3)=O)cco2)=O)CCCCC1CC1CC1 C12(CNC(c3cc(C)c(C)o3)=O)CCC1CN(C(=O)C(C(C)C)NC=O)C2 c1(COC)cccc(C(=O)NCC#CCNC(c2ccncc2Cl)=O)c1C c1(OC)cccc(O)c1CC1(C(N2CC(N3C(=O)CC(SC)C3)C2)=O)CCC1 c1(NC2CCC(N(C(C(C(C)O)(F)F)=O)C)CC2)ncnc2c1CCC2 c1(C(=O)NC(c2ccccc2F)CNC(CC)=O)cccc2c(C#N)c[nH]c12 c1(C(=O)NCC(CO)NC(C2N(CCC)CCC2)=O)cnn(C)c1N C(C(C)CN=c1cc(C)nc(-c2cccc(OC)c2)[nH]1)NC(C(C(CC)CC)C)=O C=CCCCCCC(=O)N1CC(=O)NCC1C(=O)NCCC(C)C(C)C N1(CC(=O)NC2(CN(C)C(c3cocc3Br)=O)CC2)CCSCC1 c1(C(N2CCC(NC(CCC=C)=O)C(O)C2)=O)ccc2nn[nH]c2n1 N1(C(C2CN(CCC)C(=O)C2)=O)CCCCC(NC(=O)C(F)F)C1 c1(C(N2C3CN(C(c4c(OC)cnnc4)=O)C(C3)C2)=O)c(C)ccc(C)c1C CCCCC(C(=O)N(C1CN(C(c2ccc(O)cc2)=O)CCC1C)C)C(C)C C12(CNC(CCSc3nc(C)[nH]n3)=O)CN(C(=O)CCNC(N)=O)CC1CCO2 C1(NC(Cc2c(C)n(C)nc2)=O)CCN(C(=O)CC2CC(F)C2)CCC1CO C1(C(N(CCNC(c2c(CC)scc2)=O)C)=O)CN2CCCCC2CO1 C(=O)(CS(=O)(=O)CCO)N(CCCNC(=O)CC1CCC1OC)CC N1(Cc2c(C)nc[nH]2)CCC(F)(F)C(CNC(c2ccccc2Cl)=O)C1 Cc1ccc(F)c(C(N2CC(O)(C(C)NC(=O)C(O)CC(C)(C)C)C2)=O)c1Cl N1(C(C(CC)(C)OC)=O)CCOC2(CCC(NC(c3cc(OC)ns3)=O)CC2)C1 c1(C(N2CCCC(N(C(=O)C(C)N(C)C)CC)C2)=O)c[nH]c2ncccc12 N1(C(c2onc(C)n2)=O)CCC2(CC1)CC2C(N1CCC2(CCOC2)C1)=O c1(CN2CC(C(=O)Nc3c(CC#N)cccc3)SCC2)cccc(O)c1O c1(C(=O)NC2CC(CCNC(Cc3c(C)n[nH]c3)=O)C2)ccc2c(c1)C(=O)OC2 c1(OC)cc(C(N2CC(CNC(c3ccn(C)c3)=O)CC2C)=O)nn1C O(NC(=O)C=CC(C)(C)NC(=O)CN(C(=O)COC)C)C(C(=O)OC)C C1(CC(N2C(CN(C(C3CC(O)C3)=O)C3CC3)CC3CC23)=O)(N(C)C)CCCCC1 N1(C(N2CCC(C)(COC)C2)=O)CCOC2CC(C(=O)OC(C)(C)C)CC12 N1(C(C2(C)CCCO2)=O)CC2CN(C(c3ccc(CCF)cc3)=O)CC2C1 C(C#Cc1cccc(Cl)c1Cl)NC(c1ccc2c(c1)OCO2)CC C(=O)(C1COCc2ccccc21)NCCC1(CNC(c2cc(C)oc2C)=O)CC1 c1(CC(=O)N(C)CC2N(C(Cn3c(C)ncn3)=O)CCC2)ccccc1Cl n1(CCCCNC(=O)CCn2cccc2)cc(-c2ccc(C3CC3)s2)nn1 C1(NC(C2C(SC)CCC2)=O)CCN(C(=O)CCCCN(C)C)CC(C)(C)C1 C(C)(C)(CC(=O)NCc1cccc(CNC(C2(C#N)CCCO2)=O)c1)N(C)C CC1(C(N2CC(O)C(O)C2)=O)CCN(Cc2ccc(Cl)cc2)CC1 CCCC(CC)CCC(=O)NC1(C(=O)NCc2cnn(C)c2)CCCC1 C12(CNC(C3C(=C)CC3)=O)CCCC1N(C(C1CC=CC1)=O)CCC2 C1(CC(=O)NC2(CNC(CC3C(C)(C)OCC3)=O)CCC2)COCC(C)(C)O1 CN1C(=O)OCC1C(=O)NC1C2CN(C(C3CC(Cl)(Cl)C3)=O)CC12 C1(C)(CC(=O)NCC(Cn2cc(C3(OC)CCC3)nn2)OC)CCCS1(=O)=O C1(NC(c2c(C)nc(CO)s2)=O)CCN(C(c2c(C)nc(C)n2O)=O)C1(C)C c1(C(=O)NCC(C2CCN(C(C3(SC)CC3)=O)CC2)F)ccc(C)c(Cl)c1 c1(C(N(CCC)CCN(C(=O)C(C)OC2CCCC2)CC)=O)ncn2c1CCC2 c1(C(=O)NC2CN(C(CC(=O)OC)=O)CC2C)cc(C)c2ncccc2c1C c1(C(N(CCNC(C(CSC)(C)C)=O)C)=O)cc(S(=O)(=O)N2CCSCC2)c[nH]1 c1(C(C)NCc2ccc(C(N)=O)o2)cccc(F)n1 N1(C(C(C)OC2CCCCC2)=O)CC(O)(CCNC(=O)C(Cl)=CCl)C1 c1(C(CNC(c2nc(CCOC)oc2)=O)NC(=O)C2=CCC2)ccccc1F C1(NC(c2c(CCC)cccc2)=O)CC12CCN(C(=O)CC1(C)CCOC1)CC2 N1(C(C(CCC)C(C)C)=O)CCC2CN(C(C3CC(C)OC3C)=O)CC2CC1 C(C)(C(CCC(=O)O)CCC(=O)O)NC(COCC)C(=O)OC CCC(C)(CC(=O)N1CCC(CC(C)NC(c2cc(C)no2)=O)CC1)C(=O)OC N1(C(CCc2cc(C)on2)=O)CCCC(CNC(=O)CC2CC3(CC3)CO2)CC1 N1(C(Cn2nc(C)c(Cl)c2)=O)C2CCCC1CN(C(c1cc(=O)cc[nH]1)=O)C2 c1(NC(c2nc(Nc3ncc(C(=O)OC)cn3)sc2)=O)cc(Cl)c(Br)c(Cl)c1 C(=O)(C(O)CC1CC1)NCCCOCCN(C(=O)CC(C1CCC1)C1CCC1)C C1(C(=O)NCC(C(C)C)(C)NC(=O)C2=CCCCO2)CCCC(F)(F)C1 C1(CN2CCC(c3nc(CC)[nH]n3)CC2)CC12CCOc1ccccc12 N1(C(C(=O)NCCCOC)C(C)C)CCCC(CO)(COC)C1 C(C(C(C)(C)C)NC(=O)CNC(N)=O)NC(CN(CC(=O)Nc1ccoc1)C)=O C1(C(=O)NCC2(CNC(C3(C)CC3(F)F)=O)CC2)CCCC(=O)O1 C1(CC(=O)NC2CCC(NC(C3CSCCS3)=O)CC2)CCCCCO1 CC1CC(NC(c2cnn(CC(F)(F)F)c2)=O)CN(C(C2CCCC2)=O)C1 c1(C(=O)NC2C(NC(C(c3c(C)noc3C)C)=O)COCC2)cccc(Cl)c1F N1(C(CCC)=O)CCC(C(F)CNC(c2ncoc2Br)=O)CC1 N1(C(C(S(CCC)(=O)=O)C)=O)CCc2c(CNC(=O)C(CC)SC)cccc2C1 N1(C(C2(CC)CCC2)=O)CCCCC(N(C)C(c2cc(C)cs2)=O)C1 C1(NC(C)=O)CCC(C)(CNC(=O)C(=O)N(c2cccnc2Cl)C(C)C)CC1 C1(CC)(CO)CN(C(=O)C(F)=C(C)C)C1 c1(C(=O)NCC2(NC(CCN(CCCCOC)C)=O)CCC2)n[nH]cc1[N+](=O)[O-] c1(OC)ccc(C(F)(F)C(=O)NC2CN(C(=O)C=CCN(C)C)CC2C)cc1 c1(OCC)cc(C(=O)NC(C)(CNC(=O)C(C2CCCC2)OC)CC)[nH]n1 c1(CC)n[nH]cc1C(=O)NCc1cc(C(=O)N(CCCO)CC(C)C)cs1 n1(CCNC2(c3nnnn3CCCF)CC(SC)C2)c(C)nc2ccccc12 c1(CC)nn(C)c(C(N2CCC(NC(c3cc(CC)c[nH]3)=O)C(F)C2)=O)c1Cl C1(C2(NC(C3CC3C(F)F)=O)CC2)CCCN1C(c1ccsc1)=O c1(CNC(c2cccc(Cl)c2Cl)C(=O)OC)ccc(CO)c(F)c1 c1(C(NNC(C2C(C#N)CS(=O)(=O)C2)=O)=O)cccc2c(Cl)c(Cl)sc12 Cc1nnc2n1CC(C(N1CCC(N(C)C(c3csc4nccn34)=O)C1)=O)C2 C1(CNC(=O)CC2C=CCC2)CC2CCCCC2N1C(c1ccnn1C(F)F)=O c1(NC(=O)NCc2ccc(-n3cccn3)cn2)occc1C1=CCNCC1 c1(C(=O)OCC(=O)NC2CCCN(CC)C2=O)cc(F)cc(F)c1O c1(C(N2CC(OCCNC(CNC(C)=O)=O)C2)=O)c(C)csc1Cl c1(C(N2CCC(CCNC(c3nnn(C)c3N)=O)C2)=O)ccc2c(c1)CCC=C2 c1(C(=O)OC)cc(NC(C(C)NC(C2CC(CF)C2)=O)C(C)C)ccc1[N+](=O)[O-] c1(CC(N2CCCC(C)(CNC(c3cscc3F)=O)C2)=O)ccc2c[nH]nc2c1 Cc1cc(=O)c(C(=O)N(C2CCN(C(=O)CSC3CC3)C2)CCO)cn1C1CC1 c1(C(=O)NCCCN(C(=O)C(O)C(F)F)CC)cccc(C)n1 C1(NC(c2nc(Cl)sc2Cl)=O)CN(Cc2c(Br)ccnc2Cl)CCC1(F)F c1(C(N(CC(C)NC(=O)Cc2cnc[nH]2)C)=O)ccccc1CCN(C)C CC1CCCCC1(C)C(N1CCN(C2CCN(C(=O)CCC(C)(C)C)C2)CC1)=O N1(C(c2n[nH]c(CC)c2Cl)=O)CC2CC(NC(=O)C(c3sccc3C)OC)C1C2 c1(OC(C)=O)ccc(C)cc1OCC(=O)NC1C(NC(CCCC)=O)CCC1 c1(OC)cc(F)ccc1CNC1CCCN(C(c2cncc(O)c2)=O)CC1 C1(NC(C(CC)OC)=O)CCN(C(=O)CSCc2cccnc2)CCC1CO N1(C(C2CC(C)(F)C2)=O)CCOC(CCCNC(c2n[nH]cc2Cl)=O)C1 N1(C(COCCCC)=O)CCCCCC(NC(C2CC3(C2)CC(O)C3)=O)C1 C1(C(N2CC3C(C(=O)NCC(C4CCC4)OC)(C3)C2)=O)CCCCCCC1 Cc1nccc(Br)c1NC(C1CC2(CCC2)C1)=O.c12cccnc1C(=O)N2 C1(C(N2CCC2CF)=O)C2CC3C(C2)C13.C(=O)(C(F)CC1CN(C(=O)N)C1)OC C=CCC(CC(C)C)C(=O)NC(C)(C)C(C)CC(=O)NC12CC=CC(C1)OC2 c1(C(=O)NC(CC)CNC(=O)C(C(C)(C)C)OC)c(F)ccc2c1OCO2 C(=O)(C(O)CC(F)(F)F)N1CCOCC(NC(C2(C#C)CCCC2)=O)C1 c1(SCC)ccccc1C(=O)NCC(C(C)C)NC(=O)CCCC1CC1 Cc1nnc(C(=O)NCC2CC(F)(CNC(=O)C=C3CCSCC3)C2)s1 c1(OC)ccc(CC(=O)N(CCN(C(=O)Cc2csnn2)C)C(C)C)nc1 Cc1ccc(Br)c(F)c1C(N1CCC(O)C1C(=O)Nc1c(Cl)cccc1C#N)=O CC1N(C(CCC2CC2)C(=O)NCC(F)F)CCCC12CCC2 c1(C(N)=O)ccc(C(N2CC(C(N)=O)(CNC(=O)Cc3ccc(Cl)s3)C2)=O)[nH]1 O=C(CCS(=O)(=O)C1CCC1)NC1CCC2(CC1)CC2NC(c1csnn1)=O c1(CNC(=O)C(c2cccc(F)c2Br)F)cc2c(o1)CCCC2 C1(C(N2C(C)CC(NC(C3CC34CCCC4)=O)CC2)=O)CNC(=O)CC1(C)C CCC(C)(CNC(C1CC(=C2CC2)C1)=O)C(=O)NCC1(c2ccccc2)CC1 c1(C(N(C2CCN(C(C3CCCN3C)=O)C2)C)=O)c[nH]c2cc(Br)ccc12 C(=O)(CC1=CCCC1)NC1CC(C(N(OC)C)=O)C1(C)C c1(C(=O)NC2CC(CNC(c3cc(C)nnc3)=O)C2)cc2occc2[nH]1 c1(C2(C(=O)NC(CNC(C3C(C#C)C3(C)C)=O)C)CC2)ccc(Cl)c(F)c1 CC1=C(C(=O)NC2(C(N3CC4C=CC3CC4)=O)CSC2)CCCO1 c1(C(=O)NCCC(=C)CNC(=O)CCOCC2CC2)ccncc1C(F)F c1(C(N2CC(CNC(c3nc(OC)oc3)=O)C(C)C2)=O)cc2cnn(C)c2s1 CCCC(C)(C)CC(=O)N1CC(NC(c2cc(C#N)cs2)=O)C(C)C1 c1(C(=O)NC(C(C)NC(c2c(CCC)occ2)=O)C)onc(Cl)c1C c1(SC)ccccc1NC(=O)C(CCN(C)C)NC(=O)CCc1ccn(C)n1 Cc1nc(C)c(CC(=O)NCC2(NC(c3c[nH]nc3Cl)=O)CCOC2)s1 CN1CCCCC1CC(N1CCCC1C(C)(C)CNC(=O)CSC(C)(C)C)=O C(CCN=c1[nH]cc2ccnc-2[nH]1)NC(C1C(c2cn(CC)nc2)OCC1)=O C(=O)(C(C)(C)CCCF)N1CCN(CCN(C(CN2C(C)CCC2)=O)C)CC1 C1(CC(N2CC(O)(CC)C2)=O)CN(C(C2(C(N)=O)CC2)=O)C(C)(C)C1 Cc1c(Cl)ncc(F)c1CNCc1cncc(-c2cn[nH]c2)c1 c1(C(=O)NCC=C2CCN(C(Cc3c(CC)con3)=O)CC2)[nH]c(C)cc1C C(=O)(C(O)(C(F)(F)F)C1CC1)NCCCC(C)NC(=O)CC1CN(C)CC1O C1(N(C(C=NOC)=O)C)CCCC2CN(C(=O)CSCC(C)=O)CC12 c1(C(N2CCC(CN(C(=O)C(F)(F)c3ncc[nH]3)C)C2)=O)csc2ccccc12 C(=O)(C(C(C)C)C(C)C)NC1(C(=O)NC(C(=O)OC)C)CC1 C1(C(=O)NCCCNC(CN(C)C(=O)OC(C)(C)C)=O)C2CCC12 C1(CNC(=O)Cc2ccc(C(F)F)cc2)CN(C(=O)C(O)CC2CC2)CCCO1 C1(CC(=O)NCC(CC)(C)C)CCCN(C(=O)CC2CC=CC2)CC1 N#Cc1cnc(NC(C2CC23CN(C(C2CCC(=O)N2)=O)C3)=O)c(Cl)c1 C(=O)(C(C(=O)NCC1CCCN1C(=O)CCCc1ccc(C)s1)C(C)C)OCC c1(C(=O)NC2CC(C)(NC(C(CCSC)O)=O)C2)c[nH]c2nccc(Cl)c12 N1(C(CC2(OC)CC2)=O)CC2(COC(C)C2)C1.C12CCCCC1C(=O)N2 C=C1CCN(C(c2coc(C3CC3)n2)=O)C(C(=O)NC(c2cnsc2)C)C1 C(=O)(C(Cn1ccnn1)NC(C1CC(F)(CF)C1)=O)N1CC(O)(CC=C)C1 c1(NC(C(=O)NC(CC)CCOC)=O)cc(I)c(Br)cc1C c1(C2(C(N3CC(C)OC(C)C3C)=O)CC2)cccc2c1OCCO2 Cc1cc(=O)n(C)cc1C(N1CCC(NC(=O)C2=COCCC2)C(C)(C)C1)=O Cc1cc(=NC(=O)C(=O)N2CC(F)(F)CC2(C)CNC(=O)CNC(N)=O)[nH]o1 c1(C(N(C)CC2CCN(C(c3c(C)onc3)=O)C2)=O)nccc2c1CNC2=O c1(OCCC(=O)NC2(C)CCN(C(=O)CC3(OC)CC3)C2)ccc2c(c1)CCC2 C(C)(CO)(C(=O)N(CCCC(C)(C)NC(c1[nH]c(C)cc1C)=O)C(C)C)NC(C)=O C1(C(N2CCCC(NC(C3CC4CCC(C3)C4)=O)C2)=O)CC2(C1)CC2(F)F Cc1cc(O)cc(O)c1C(=O)NC1(CNC(C2CCCCO2)=O)COC1 C1(C(N(CC(C)NC(=O)CCCNC(=O)C2CC2)CC)=O)(SC)CCC(F)(F)C1 C(=O)(C1=CCCCC1)N1CCC(C(C)NC(CC(=O)N(C)C)=O)CC1 CCC(C)(C)C(O)C(=O)NC1CCC12CN(C(c1cccc(OC)c1N)=O)C2 CCCS(=O)(=O)CC(=O)NC1CC(OC)CN(C(=O)CN2CCC(F)(F)C2)C1 C1(CC(=O)NCC(C)N(C)C(C2CC23CC(O)C3)=O)CCCOCC1 C(=O)(C(O)CC(C)C)NCC(CO)NC(Cc1c(C)nc(C2CC2)s1)=O N1(C(c2ccc(CC)nc2)=O)CCCC(NC(=O)CCC2CCCO2)C1CC N1(C(Cn2cnc(C#N)n2)=O)CCC2CN(C(C3(c4cccs4)CC3)=O)C2C1 c1(C(=O)NCC2(O)CCCN(C(=O)CNc3nccs3)C2)ncnc2c1CCCC2 CC1CC(C(=O)NC2CCCCN(C(c3ccc(CF)cc3)=O)C2)=NO1 Cc1cocc1C(=O)NCC(C)CNC(c1c[nH]nc1-c1ccsc1)=O CC(CC(C)NC(c1c[nH]nc1I)=O)NC(=O)C(=O)N(C)C c1(C(=O)NC2CC(NC(CC3C=NN(C)C3=O)=O)C(O)C2)cccc(Cl)c1O C(=O)(C#CC(C)(C)CNC(=O)C=CC(=O)N(C)C)N1C(C(C)C)(CO)CC1 c1(CC(=O)N(C2(C)CCN(c3ccnc(Cl)n3)C2)C2CC2)c[nH]c2ccccc12 N1(C(C2CC(N(C)CC)C2)=O)CCOC(C)(CNC(=O)C2CC2)C1 C1(N(C(C=CCOC)=O)C)CN(C(c2cn(C3CCOCC3)nn2)=O)CC12CC2 c1(OC)cc(C)ccc1C(C)Nc1nccc(N(C)CC2CC2)n1 CCC(CC)C(C)C(=O)NCC(C)(C)CNC(C1CCC(O)CN1C)=O c1(C(N2CC3C(CN(C(C=CC(CC)=CC)=O)C)C3C2)=O)cc2ncccc2o1 C1(C)(NC(C(COC)OC)=O)CCN(C(=O)C=Cc2ccnn2C)CC1 C12CCC(C1)C(=O)NC2.c1(CCS)ccccc1.C1(C(=O)OC)(OCC(=O)N)CC1 C12(C(N(CCCCCNC(CC)=O)C)=O)CCCC(C(=O)OCC)(COC1)C2 C(=O)(C1=CC2C=CC(C1)C2)NCC(C)(C1CC1)NC(c1c(Cl)ccc(C)c1)=O C1(C)(CC)CC(NC(=O)CCCn2cncn2)CN1C(=O)C=Cc1ccncn1 c1(C2C(C(=O)NC(C(C)(C)NC(c3nc(SC)oc3)=O)C)C2)ccc(C)nc1 c1(-c2n(CC3C(C)C3)c(N3CC4CCC(CC4)C3)nn2)cccc2cc(F)ccc12 c1(C(N2CC(CCNC(C(CCOC)OC)=O)C2)=O)cc(Cl)c(F)cc1F N1(C(C2CCC(CC)O2)=O)CC(C)CC1C(=O)NCCCN1CCOC1=O C1(NC(C2CCCOC2C(=O)O)=O)CNCC(F)(F)C1 N1(C(C)(C)C)CCN(C(=O)N(c2cccnc2)C2COC2)CC1 c1(C(=O)NCC2(O)CC(NC(C(C(C)(C)C)O)=O)C2)ccc2c(n1)CCCC2 c1(C(N2CCC(NC(c3conc3C3CC3)=O)CC2)=O)c[nH]c2c(F)cccc12 c1(CNC(C(C2CCN(C(c3cc(C)sn3)=O)C2)F)=O)ccc(F)cc1C N1(C(C2(CNC(C(C)OCC=C)=O)CCOCC2)=O)CCCC(O)(CC#C)C1 N1(C(CSCCCC)=O)CC2(CCN(C(c3ncc(F)cn3)=O)CC2)CC1C CCCC(CC(=O)Nc1ccccc1C)NC(=O)CC1(COC)CC1 N1(C(Cn2ncc(C#C)c2)=O)CCC(C)(C(N2CCC(c3cc[nH]n3)C2)=O)CC1 c1(CC(=O)NC(Cn2cc(C(C)OC)nn2)C)cc(C)ccc1C O=C(C1CCSc2ccccc21)NCC1CN(C(C23CCC(CC2)C3)=O)CCO1 c1(CC(=O)NCC(CCCC)NC(=O)C(C)C)cnc(Cl)cc1N n1(CC)cc(CN2CCC3C(O)C(C)(C)C23)c2ccccc12 C1(C(=O)NCCC(C)NC(C2(c3ccno3)CC2)=O)CCN(C)CC1 CC(C)C(O)CC(=O)NCCCCC1CCN(C(C2(C)CCCC2O)=O)CC1 c1(N2CC(C(N3C(CC(=O)NCCCC)CCC3)=O)C2)nc2ccccc2s1 CN1C(=O)NC(C)(CCNC(c2ccc(OCCF)cc2)=O)C1=O C1(Cn2cc(C(CC)(C)O)nn2)C(C2CC2)CCN1C(=O)CCSC(F)(F)F NS(=O)(=O)c1cc(-c2cn(CCCN3CC4C(C(=O)O)C4C3)nn2)c(O)cc1Cl c1(C(=O)NCC2CC(C)N(C(=O)CCC#N)C2)cccc2nccn12 N1(C(c2c(C)cccn2)=O)CCC(CNC(C2COCC2C(N)=O)=O)C12CCC2 C1(NC(c2cccc(CCC)c2)=O)COCCN(C(C2(C(=O)C3CC3)CC2)=O)C1 c1(C(=O)NC2(CNC(=O)CC3CCC(=O)N3)CC2)[nH]nc2ncnc(O)c12 c1(C(N2CC(NC(c3cnns3)=O)CC3(C2)CC3)=O)ccc2c(c1)CCC=C2 N=c1ncc(-c2cn(C3CCN(c4cccnn4)C3)nn2)c[nH]1 C(N=c1cc(C)nc(-c2ccc(Br)cc2C)[nH]1)c1scc(C)n1 Cn1c(=O)sc2cc(C(N3CCC(CC4(C)CC4)C3)C(=O)NC3CC3)ccc12 N1(C(c2cc(C3CCC3)no2)=O)CC(C2CCN(C(C3CC4CC3C4)=O)CC2)C1 C1(N(C(=O)CCC2CCC(=O)N2)C)CC2CCC(C1)N2C(=O)CSC(F)F N1(C(CCCCC#C)=O)CC(CNC(=O)C=C2CCCCC2)C2CCCCC12 C(c1nc(C)c(C)[nH]1)=CC(=O)NCC1CC(CNC(C2CC(C#C)(O)C2)=O)OC1 C1(NC(C2(NC(c3cccc(CC)c3F)=O)CC2)=O)CCn2nnnc2C1 c1(C(=O)NCC(CO)NC(CCCc2n(C)cnn2)=O)cc(Cl)c(Cl)[nH]1 C12(NC(C3(COC)CN(C(C4(C)CCC(=O)CC4)=O)C3)=O)CCCN(CCC1)C2 CC(CC(=O)NC1CC(F)CN(C(=O)CCc2cc(F)ccc2F)C1)C(F)F C(=O)(C1=CCCCC1)N1C(c2ccccc2)(C(=O)NC2CC(C#C)C2)CCC1 C=CC(O)C(C)(C)C(=O)N1CCC(O)C(C(=O)N(C(C)C(=O)NC)CC)C1 c1(C(N2CC(NC(C(CC)OC)=O)C3(C2)CC3)=O)ccc(SCC)c([N+](=O)[O-])c1 C(=O)(C1=CC2C=CC1C2)N1CCC(C(C)NC(=O)CC2(C)CC2(F)Cl)CC1 CCCCC(C)C(C(=O)NCC(F)F)N1CCOC(COC)C1 C(=O)(C1=NNC(=O)CC1)NCC1CC(NC(c2c(N)non2)=O)C(O)C1 c1(C(=O)NC(C(C)NC(=O)C(N)=O)CCc2ccccc2)cc2cccnn2n1 CCCCCCC(CC)(CC)C(=O)OCC1CCNC(=O)CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(C2C(C)C2)=O)CC1N=[N+]=[N-] C1(CNC(C(C)N(C)C)=O)CN(C(c2ccc(C(C)O)cc2)=O)CCCO1 Cc1cc(F)ccc1C(F)(F)C(=O)NCCC(C)NC(c1cc(CF)on1)=O c1(CN(C(=O)CCC2CCN(C(C3CCCCC3)=O)CC2)C)nc([N+](=O)[O-])n[nH]1 c1(C(N2C(CNC(C(N)=O)=O)C=CC2)=O)ccc2c(c1)OCC2 N1(C(C#CC(C)C)=O)CCC2(CCCCC2NC(c2cc[nH]n2)=O)C1 N1(C(c2c(CC)noc2)=O)CCCC1C1CCCN1C(c1cc(F)ccc1Cl)=O c1(NCCCN2CCN(C(COC)COC)CC2)ccc2c(c1)nc(C)n2C C(CNC(=O)C(=O)Nc1ncc[nH]1)(CC(C)C)NC(CC=CC)=O N1(C(c2cc(CC)nc(Cl)c2)=O)CC2CC1CCC2NC(C1CCCC(C)C1)=O c1(NC(c2cc(CC)nn2C)=O)sc(C)c(C)c1C(=O)NCc1ccsc1COC C12(NC(c3n[nH]cc3Cl)=O)CCCC1CN(C(=O)COC1(C(=O)OCC)CC1)C2 n1(CC)cnc(C(=O)N(C)CCOCCCO)c1.C1CC(=O)N1C(C)C CC1CN(C(=O)C=Cc2ccco2)CCC1Nc1cc(=O)n(C)cn1 N1(C(Cc2nc(C(C)(C)C)sc2)=O)CC(NC(=O)C(Cl)=CCl)C2(CCC2)C1 c1(C(N(CCNC(=O)C(CO)N(C)C)CC)=O)nc(C)c(=O)[nH]c1N c1(C(=O)NC2CCN(C(c3c(C)c(Br)no3)=O)C2)cc2c(nn1)CCCC2 N1(C(c2ccc(C(C)=O)s2)=O)CCC(O)(CN(C)C(c2ncn(C)n2)=O)CC1 C1(CNC(C=CCCC)=O)CC2(CC2)CN1C(C1C2CC3C(C2=O)C13)=O N1(C(c2c(O)ccc(N)c2)=O)CC2(CCCC2NC(=O)CC2CSCCS2)C1 N1(C(CC2(CNC(C3CC3(Cl)C(=O)O)=O)CC2)=O)CC(C=C)(CC=C)C1 Cc1ccccc1CN1CCN(C(=O)C(=O)NC(C2CC=CCC2)C)CC1 N12CC(C1(C)C)CN(C=O)CCC2=O.c1(CC=CC)c[nH]c(=N)o1.OC c1(CC(=O)NCCC(C)NC(COC)=O)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NC(C(N2C(C)(C(C)C)CC2)=O)CC2CCCC2)CC2(CC(=O)C2)C1 c1(CCC(=O)NC(C)CNC(C23CCOCC2C3)=O)cc2ccccc2[nH]1 C(=O)(C(F)C(C)C)N(C(CNC(c1ccn(CCCC)n1)=O)C)CC C1(CNC(C2C3COCC23)=O)CC2(CCC2)CN1c1cnc(F)cn1 C(=O)(C1=NOCC1)NCC1C(CNC(=O)CCSc2ccccc2)C1.CSC c1(C(N(CC(C)N(C(C(C(C)C)n2cc(C)nc2)=O)C)C)=O)cc(C)nc(C)c1 C=CCCCC(C)NC(=O)C(CCOCC)NC(c1cnnn1CC)=O c1(NC(=O)CNC(=O)NC(C2CCCC2)=O)cccc(Br)c1Cl Cc1cc(C(N2CCOC(C(C)NC(=O)CNS(=O)(=O)C3CC3)C2)=O)cn1C N1(C(c2cc(C)cc(F)c2)=O)CCCC(NC(c2ccn(C)c(=O)c2)=O)C(F)C1 N1(CC(=O)NCC(C(C)C)=O)C(C)(C)CC(=O)CC1(C)C.n12cc(nn1)CC2C C12(NC(=O)COc3cccc(F)c3)COCCC1CN(C(c1nsnc1O)=O)C2 C=C=CCCC(=O)NCC1CCCN(C(=O)C(C)(C)c2cncs2)C1 N1(C(=O)CCC2CCCC2)CC2CC(C1)CN(C(=O)CCc1ccc(O)nn1)C2 C1(C)(CC)C=C(C(=O)OCCC(=O)NC(C2CCCCC2)(C)C)C1.C1(O)CCCOC1 Cc1nsc(N)c1-c1cn(CCC(=O)N(C2CC2)CC2(C3CC3)CCCO2)nn1 C1(NC(=O)CC2C=CCCC2)CCC(O)CN(C(c2csc(C3CC3)n2)=O)C1 C12(C(N3CCC(C)C(N(C(=O)C=Cc4ccsc4)C)C3)=O)CCC(CC1)C2(C)C c1(N2C(=O)CC(NC(=O)NC(c3nccn3C)CC)C2)ccc(C)c([N+](=O)[O-])c1 C1(NC(CN(C2CC2)CC)=O)C(C)CN(C(C2(OC)CCC2)=O)CC1C C=C(C)C1OCCCC1C(=O)NCCC(C)N(C(=O)CC12CCC(CC1)CC2)C C1(N(c2cnc(C)s2)C(C(c2ccccc2)OC)=O)CCCC12CCNCC2 N1(C(C)=O)CCC2(CCCN(C(=O)CNC(c3cnc(O)nc3O)=O)C2)C1 Cc1ccc(F)c2oc(C(=O)NCCC3CC(C)(C)NC3=O)cc12 C(=O)(C(C)(C)CC1CCOCC1)N1CC(O)(CNC(CC2C(C)OCC2)=O)C1 S(=O)(=O)(c1cccc(N2CCSC3(CCOCC3)C2)n1)N(C)CC1CCN(C)C1 C(=O)(C(F)(F)CSc1ccccc1)NCC(CNC(=O)CCC1(C)CC1)OC CN1CCCC12CCN(C(C1CC(F)CN1C(C1CCCO1)=O)=O)C2 c1(OC)ccc2nc(COC3CCCNC3)[nH]c(=NCCN3CCC3)c2c1 c1(CC)nn(C)c(CC)c1C(=O)NC1CCCC1NC(=O)CC1CCN(C)C1 CCCC(CCCNC(=O)C(CC)n1cccn1)NC(c1ccc(Br)cc1C)=O N1(C(CSC)=O)CCCC(C)C1CNC(=O)C(C)(C)OC.c1(O)cc(F)cc(Cl)c1 Cc1nc(NCC2CC(C)(C)CCO2)cc(NC2CC2C2CCC2)n1 C(C(=O)N1CCCc2nccn21)CCO.CC(C)(C(=O)CCN)C1CCCC1.O N1(C(CSCC)=O)CCN(C(=O)C(Cc2ccccc2)N(C)C)C2CCC12 N1(CC(=O)Nc2cc(C)cc(C)c2)CCOCC1C1CCCO1 c1(C(N2C(C)CCC(NC(CC=CC)=O)C2)=O)cc2c(nc1O)CCC(C)(C)C2 C(=O)(C1=COc2ccccc2O1)NC1CC(C)(NC(C(CCC)O)=O)C1 N1(C(C(N2CC(CC)(CN)OCC2)=O)=O)CCn2c(nc(C(F)(F)F)c2OC)C1 N1(C(c2c(C)ccc(F)c2)=O)CCC(NC(C2(F)CCOC2)=O)CC(C)(C)C1 CCC(CN(C)C)CC(=O)N(C(CNC(=O)Cc1nccn1C)C1CC1)C N1(C(c2cnc(C)nc2)=O)CCOC2CN(C(=O)C(C)O)CC12 CC1(CNC(C2CNC(=O)C2)=O)CCCN1C(c1ccsc1-n1cnnn1)=O Cc1cccc(C(=O)NCC(N2CCN(C(=O)CSC3CC3)CC2)C(F)F)c1O N1(C(C(C=C=C)C)=O)CC(=O)NC2CN(C(=O)Cc3c[nH]nc3C)CCC12 C1(CCNC(CCCNC(=O)OC)=O)(NC(c2cscc2Cl)=O)CCOCC1 N1(C(CC)=O)CC(C(=O)O)C2(C1)CN(C(=O)CCc1c(OC)cccc1C)C2 C1(CNC(C2=NOC(C)C2C)=O)CC2(CCOCC2)CN1C(c1nccn1C)=O C1(C)(C(=O)NCC(COC)NC(C23CCCN2CCC3)=O)CCCCCC1 c1(-c2n(-c3ccc(Cl)nc3)nc(C3CCCC3)n2)n[nH]c2ccc(I)cc12 CC1(C)COC(CC(N2CC(O)(CNC(=O)CCN3CCC3)C2)=O)C1 c1(C(N2C(CO)CC(NC(c3cn(CCC)nc3)=O)C2)=O)ccc(C#N)cc1C C1(CC#N)CCCCC1NC(c1cnc(CNC(=O)C=Cc2cnc[nH]2)nc1)=O c1(C(=O)NCC(CNC(c2cnn(CC)n2)=O)(C)C)cccn2c(C)nnc12 c1(COCC)cncc(C(N2CC(O)(C(F)C(=O)Nc3[nH]c(C)nc3C)C2)=O)c1 N1(C(CN(CCC)C)=O)CCC(NC(=O)C(C)(C)C2CCCO2)C(CC)C1 C1(NC(C(c2cccc(OC)c2)(C)C)=O)CN(C(=O)CSC(F)F)CC12CC2 C=CCC(CC(C)C)C(=O)NC1(c2ccccc2)CCN(C(C2CC(F)C2)=O)C1 CCC(C)C(C(=O)N1CC2(CC(CNC(=O)C=CC(C)(C)C)C2)C1)NC(N)=O.OCC c1(C(N2CC(NC(Cn3c(C)cc(C)n3)=O)C3(C2)CC3)=O)ccc2c(c1)CCO2 c1(OC)ncccc1C(=O)NC(C)(C)C(=O)NCCN(C)C CCC(F)(F)C(C)(C)C(=O)NC1CCC1CNC(c1[nH]cc2c1CCS2(=O)=O)=O Cn1ncc(C(=O)NCC(C2(O)CN(C(=O)CCc3cc(Cl)no3)C2)(C)C)n1 C1(NC(c2c(C)cco2)=O)C2CCC1CN(C(=O)Cc1sccc1C)C2 C1(CC(N2CC(CC(C(=O)NCC(C#C)CC)F)C2)=O)CCCN(C)C1 c1(C(N2CCCC(NC(C3(N(C)C)CC3)=O)CCC2)=O)nc2cc(F)ccc2s1 c1(C(=O)NC2CCN(C(CC(C)(C)C)=O)CC2(C)C)ccc(F)c(F)c1O C1(CC(N2C3C(NC(c4c(C)nc(C)[nH]4)=O)CC(C3)C2)=O)CCC2(CCC2)CO1 O=S(=O)(c1ccc(NCCCOC(=N)O)cc1Cl)NCC(c1ccc(F)cc1)CO c1(C(=O)NCCCN(C(C(COC)(C)O)=O)C)csc2nnsc12 N1(C(C(CC#C)(C)NC(C2C(C#N)C2(C)C)=O)=O)CCC2(CCSC2)C1 c1(CC(=O)NC23CC(CNC(c4ccc(C)s4)=O)(OC2)C3)c(C)cccc1C Cc1cc(C)c(C(N2CCC(O)(CCNC(c3coc(Cl)n3)=O)CC2)=O)cn1 CC1CN2CCCCC2CN1C(=O)CCc1cccc(F)c1Cl C1(C(=O)NCC=CCNC(C2CC2F)=O)CCc2c[nH]nc2C1 CCCCC(C(=O)NCC(CC)NC(=O)CC1C=NN(C)C1=O)C(C)C C1(NC(C(N(C(C(C)=C2CC2)=O)C)C2CC2)=O)CNC(=O)C1(C)C N#CC1CN(C(C2CCCCO2)=O)CCN1C(c1cocn1)=O C(=O)(CCS(=O)(=O)N1CCOCC1)N1CC(NC(C(C=C=C)C)=O)C(O)C1 c1(CC(=O)NC2CCC23CN(C(c2nn[nH]c2Cl)=O)C3)ccc2cc[nH]c2c1 CCCC(C1CC1)NC(=O)N(CCC)C(C1CC1)C1CC1 CCC(CCOC)C(=O)N1CCCC(C(=O)Nc2cccc(F)c2OC)C1 c1(SCC(=O)NC(CNC(C(c2ccc(OC)cc2)C)=O)C)cc(C)ccc1C C=C=CCCC(=O)NCCOC(C)(C)CNC(C1(CNOCC)CCCCC1)=O C1(C(C)NC(C2(CN(C)C)CC2)=O)CCN(C(=O)CCc2cnoc2)CC1 N1(C(c2c(C)snc2)=O)CC2CC1CC2NC(=O)Cc1ccc(Br)nc1 C(=O)(C1=CC2CCC=CCCC12)NCC1N(C)CCN(C(C2CNC(=O)N2)=O)C1 c1(C(N2CCC(O)(CO)CC2)=O)cnc2n[nH]c(C3=COCCC3)c2c1 c1(C)cncc(N)n1.CCC(C(=O)N1CCCCC1)N(CC)CC.N12CCC1C2=O c1(C(=O)NCCCCN(C)C(C23CC(F)(C2)C3)=O)cnc2sccn12 C(=O)(CCCC(CC)CC)N(C(C(N1CCC(OCC=C)C1)=O)(C)C1CC1)C C1(NC(CC2C(NC(C(C)(C)n3ccnn3)=O)CCO2)=O)CCCC2(CCC2)C1 C1(NC(C2(C(F)F)CC2)=O)CCCC1C(N1CCC(C(C)N(C)C)C1)=O c1(CC(N2CC(C3(NC(C(C=C)O)=O)CC3)C2)=O)cc(F)cc2c1OCOC2 C(C(C(=O)NOC1(OC)CC1)NC(=O)CC1(OC)CCC1)OCC c1(C(=O)NCCCCNC(C(C)NC(=O)C(C)(C)C)=O)cnn(C)c1S(N)(=O)=O c1(C(N2CC(C(N)=O)(CNC(C(CC)SC)=O)C2)=O)cncn(C)c1=O c12ccc(cn1)-c1cn(nn1)C2.C1(CC(=O)OC)CCCCO1.C12CC(C1)NC2 Brc1ccc2c(c1)CCC(Oc1ncsc1Br)O2 N1(Cc2ncn(C)n2)CC(NC(c2cc(Cl)cc(Br)c2)=O)C(F)(F)C1 C(=O)(C1=NOC(CNC(=O)C=C(C)c2ccco2)C1)N(C1CCCC1)CC N1(Cc2c(CC)onc2C)CC2CC1CN2C(c1coc(C(C)C)n1)=O C(=O)(C1CCCc2nccn21)NCC1(C)CCCN(C(c2cnnc(O)c2)=O)C1 C1(CC(=O)NCCC2(O)CN(C(=O)CCc3nc(O)n[nH]3)C2)C=CS(=O)(=O)C1 Cc1ccc(C(N2CCCN(C(c3csc(C)c3N)=O)CC2)=O)cc1Cl CC(C)(C)CC(F)C(=O)N1CCC(C)(NC(=O)C(F)=CCOC(C)(C)C)C1 CC1CC(C(N2CC(CF)C2)=O)N1C(c1ccoc1)=O S(=O)(=O)(c1[nH]c(=NC2CCC(=O)NC2)ccc1Br)N1CCC(C)(F)C1 C#Cc1cc(C(=O)COC(C2C3CCC(C3)C2OC)=O)cc(F)c1 C(=O)(C(CNC(C1CC=C(C)CC1)=O)C(C)(C)C)NCCS(CC)(=O)=O C1(CC(=O)N(CCCCCNC(c2cc(CCOC)on2)=O)C)CCC2CC2C1 CC1(C)CN(C(c2cc(C(F)F)[nH]n2)=O)CC1CNC(C1CCCC(F)(F)C1)=O CC(CC(=O)N(CC(C)CNC(C1CCCS1)=O)C)N(C)C C1(N(C)C)CCC(C(N2CC(F)(C(=O)NOCC(C)(C)O)C2)=O)C1 c1(CC(=O)NC(C2CCCCC2)CNC(c2cnc(SC)s2)=O)cnn(C)c1C C12(C(N3C4(C(=O)NCCC(C)CO)CC4CC3)=O)CCC(CC1)CC2 n1(CC(=O)NCC2CN(C(C(C)C)=O)C(C)(C)C2)nc2n(c1=O)CCCCC2 N(C(=NCCF)N1CCC(CC(=O)OC(C)(C)C)C1)CC(CS(CC)(=O)=O)(C)C CC1CC(CNC(=O)C(C)(C)F)CCN1C(c1cc(N)cn1C)=O c1(C(=O)NCC(CNC(C(F)OC)=O)CO)ccc(C(F)(F)F)c(F)c1 N1(C(C(C)c2ccsc2)=O)CC(C)(NC(c2cc(C3CC3)on2)=O)C1 C=C(C)C(CC(=O)N1CCOC(CN(C)C(c2cnccc2Cl)=O)C1)OCC N1(C(CCCCOC)=O)CCCC(C)(CNC(c2c(OC)cccc2F)=O)C1 N1(C(c2cc(COC)no2)C(=O)NC)CCOC(CF)C1(C)C c1(C(N2CC(NC(C=CC(CC)=CC)=O)CC2(C)C)=O)cc(S(N)(=O)=O)oc1Cl N1(C(C(C)OCCCC)=O)CCC(CO)C(NC(c2nn(CC)cc2Cl)=O)C1 C1(OC)CCCC(C2CC(C)C2)C1.C1C(=O)N1.C(=O)(CNC(=O)OC(C)(C)C)N C1(CNC(C2(C(C)C)COC2)=O)COCCN1Cc1cn(CC(=O)N(C)C)nn1 N1(C(C(Cc2ccccc2)ON)=O)C2CCC1CC(=O)NC2 CC(CC(=O)NC(C)(CNC(=O)C=CC=C(Cl)Cl)CO)N(C)C c1(C(=O)NCC2CCCN(C(C(C(C)C)(C)O)=O)C2)ccc(P(C)(C)=O)nc1 C(=O)(C(C)C(O)CCCC)NC1C(C(N2CC(C#C)C(OC)C2)=O)CC1 c1(C(N(CC(C)NC(=O)C(C)(C)C)C(c2cnccn2)=O)=O)cnc(Cl)cc1N N1(C(C(C)S(C)(=O)=O)=O)CC2(CCN(C(=O)CCCN=[N+]=[N-])C2)C1 c1(C(N2C(CNC(CC3(OC)CC3)=O)C(C)CC2)=O)cc(Br)cnc1C O=C(C(O)C1=CCCCC1)NC1(C(N2CC3CCC2C3)=O)CCSC1 N1(C(C(CC)N(C)C)=O)CCC(C)N(C(=O)COc2ccc(NC(C)=O)cc2)CC1 C1(CC=C)(NC(=O)Cc2nc[nH]n2)CCN(C(c2ccc(OCC)nc2)=O)C1 N1(C(c2nccc(C)n2)=O)CCN(C)CC1CNC(=O)CC1(O)CCCCC1 CC1CN(C(=O)Cc2cscn2)CCN1Cc1cc(O)ccc1Br c1(C(=O)NCCN(C(=O)CC2CCSCC2)C(C)C)csc(CO)n1 Cc1c(C(=O)NCCCNC(C2CN(C)CC2C)=O)cc(F)cc1[N+](=O)[O-] N1(C(c2c(C)noc2)=O)CC2CCC1CN2C(=O)C(C)CO C1(NC(CC=CC)=O)CC12CCN(C(=O)CCn1ccc(O)nc1=O)CC2 c1(CC(C(=O)N2CC(N(C(C(C)OCCCC)=O)CC)C2)C)ccc(OC)cc1 N1(C(c2cnc(C(C)C)o2)=O)CCOCC1C(=O)NC1(CCN(C)C)CCC1 Cc1cccc(N)c1C(=O)NC1CCN(C(C2(n3cccn3)CCC2)=O)C1 C1(NC(C(c2n(C)ccc2)=O)=O)COC2(CCCN(C(=O)C=C3CCC3)C2)C1 C1(N(C(C(c2ccccc2)SC)=O)C)CC2CCC(C1)N2C(=O)C1=CCSC1 CCC(C#N)C(=O)N1CC(N(C)C(c2nn(C)cc2C)=O)C1 Cc1cc(F)c2cc(C(=O)NC3CC(NC(c4cc(Cl)ccc4N)=O)C3)[nH]c2c1 N1(C(C2(NC(C)C)CC2)=O)CCCN(CCNC(c2cocc2C(N)=O)=O)CC1 c1(C(N(CCNC(c2c(C)csc2)=O)C2CC2)=O)cc(N)ccc1Br N1(C(c2c(C)cc(Br)cc2F)=O)CCc2c(C(=O)NC(C)CO)csc2C1 Cc1nnccc1C(N1CCCCC1CCNC(=O)CC1CN(C)C1)=O c1(C(C(=O)NCC(=C)C)N(C(C)Cc2ccc(C)s2)C)ccc(N(C)C)cc1 n1(C(CC)C)nnnc1C(c1cnoc1C)NCc1cncs1 c1(N(C(c2c(CC)scn2)=O)C)cc(C2CC2)ncn1.C12CCCN1C2 c1(C(=O)NC23CC(NC(c4cc(C(C)=O)cn4C)=O)(C2)C3)ccc2cnnn2c1 C1(c2n(C)ncc2)CCC2(CC1)CC2C(=O)N(CC1(O)COC1)CO.C(=O)(C1CC1)N N1(CCNC(=O)CSc2cccs2)CCN(C(=O)C(c2nc(C)cs2)C)CC1.CO c1(C(=O)NC(CCN(C(C(CC)OC)=O)C)C(C)(C)C)cn2cc(C)sc2n1 C1(NC(C2CCN(C(C3C(OC)CC=CC3)=O)CC2)=O)CN2CCCC1C2 c1(CC(=O)NC(CNC(c2ccc(OC)cc2)=O)C)cccc(Cl)c1OC C(=O)(CC(C)(O)COCC)N1CCCC(CC(=O)NCC(COCC)C)C1 CCCC(C#N)C(=O)N1CCCC(CNC(=O)CCn2ccccc2=O)CC1 C1(NC(CCOCCCNC(C2C(C)CCCC2)=O)=O)CC2CC1CC21CC1 C1(C(=O)NCCc2cc(C)on2)CC12CCN(C(c1ccncc1)=O)C2 C1(C(N2CCC(C(C)C(=O)N(CCO)CCO)CC2)=O)CCC=CCCC1 Cc1ccc(OCC(=O)NCC2CC(F)(F)CN2C(=O)CCC2CC2)c(C)c1 C1(c2ccc(CC)s2)CN(Cc2ccc(OCC(=O)O)cc2)CCO1 C=C(C)CCCC(=O)N1CCCCCC1CNC(=O)C(c1c(C)cccc1C)O N1(C(C=C(C)C(F)F)=O)CCOC(CN(C(=O)CC2CCC3CC23)C)C1 Nc1c(C(=O)NC2CC(CCNC(=O)C(F)(F)C(O)C3CC3)C2)cc(F)cc1F C(c1ccc(Cl)c(Cl)c1)=CC(N1CCC(CNCc2cnc(Cl)s2)C1)=O Cc1cnn(C)c1CN(C)C(=O)NCC(C)(CO)c1ccccc1 Cc1c(C(=O)NCC2CCN2C(c2nn(C)cc2[N+](=O)[O-])=O)sc2cncn12 C1(F)(CNC(c2n3cc(C)sc3nc2)=O)CC2CCC(C1)N2C(=O)C=CBr C(=O)(C(O)CCS(C)=O)NC1CC(C)(NC(c2cnc(-c3cccc(C)c3)s2)=O)C1 C1(C(=O)NC(C2CCCCC2)CNC(C2C(C#C)CC2)=O)CCn2ncnc2C1 c1(C(=O)NCCC(C)NC(C2(N(C)C)CCCCC2)=O)cc(O)cc(Br)c1 C(=O)(C1COc2ccc(Br)cc21)NC1(C)CCN(C(C2(C#C)CCC2)=O)C1 C(C1CCCN1C)=CC(=O)NCC(CN(C(=O)CC1CCCC1)C)O N1(c2c(OC(C3C(C(=O)OC)CC=CC3)=O)nccn2)CCCN(CO)C(=O)C1 CN1CCCC2C(C(=O)NCC3CCCC(C)(C)C3)C1CCN2 c1(NC2CCCN(Cc3nc(C)on3)C2)nccc(C)c1C#N C1(NC(c2cnn(CCNC(=O)Cn3ccnn3)c2)=O)CCOCC1F C(C(C(=O)N(C1(C)CC1)C)C(C)(C)C)NC(CCCOC(C)C)=O c1(-c2c(C)c(F)c(F)cc2)cccc2c1CNS(=O)(=O)O2 C#Cc1ccc(C(=O)NCCC2CN(C(=O)CN(C)C(C)=O)CCCO2)c(F)c1 n1(CC(=O)NCC2CCN(C(C3C(COCC)C3)=O)CC2)cc(S(N)(=O)=O)cn1 c1(C(N2CC3C(NC(C4C(C)(C)COCC4)=O)(C3)C2)=O)csc(S(N)(=O)=O)c1 C(=O)(CCCC(F)(F)F)NC(CCOC)CNC(C1CCC=CCCC1)=O Cc1ccsc1C=CC(=O)NCC1CCC1NC(=O)C(C)C1CC1 C1(OC)CC(C)N(C(c2cnn(-c3ccc(Cl)cc3)c2)=O)CC1C C1(C2CCN(C(=O)CC3CCCCC3O)C2)(NC(C2CCCO2)=O)CC1 c1(CCC)ccccc1C(=O)N(C1CN(C(=O)COc2ccccc2CC)C1)C c1(OC)cc(C(N2CCC(NC(c3cnc(Cl)cc3Cl)=O)C(O)C2)=O)ccc1Br N1(C(CNC(c2c(C)occ2)=O)=O)CCN(C(=O)CC2(C)CCCC2)C2(CC2)C1 CCCCCCC(C)C(=O)N1CCC(NC(=O)CN(S(=O)(=O)CC)C)C1 C(=O)(CCCC(C)(C)CC)NCCC1CC(NC(c2n(CC)cnn2)=O)C1 CC1CN(C(=O)COC2CCC2)CC(C)N(C(c2cscn2)=O)C1 CC1(C)CC(CNC(C2(C)CCCS2)=O)CN1C(=O)CCC1CCCCC1 C1(CC)C(C(=O)NC(C)Cc2nc[nH]n2)CCCN1C(c1coc(C)n1)=O CCCCCC(C)CC(=O)N1C2CCC1CN(C(=O)Cn1nnc(=N)[nH]1)C2 c1(C(N2CC(NC(c3cncc(C)c3)=O)C3C2C3)=O)cc(N)nc(Cl)c1 CCC(CC(F)(F)F)C(=O)NC(CNC(=O)CC1CCC1)C1CCC1 C=C1c2ccccc2C(=O)N1C(C)C(=O)OCC1OCCC12CCC2 Cc1c[nH]c2ncc(C(N3CC=CC3CNC(=O)C(C)C3CCC3)=O)cc12 CN1C(=O)CSC1=CC(=O)NCCOCCCNC(=O)COC1CC1(F)F C1(NC(CC=C)=O)CCOC1C(=O)NCC(C)Cc1cn[nH]c1 C12(CCNC(Cc3scc(C)c3)=O)CCC1CN(C(C1(C)CS(=O)(=O)C1)=O)C2 c1(-c2cn(CCN(C(=O)CC3CCC(C(F)(F)F)O3)C)nn2)cccc(C#N)c1 C(=O)(C(COC)NC(C)=O)NC(COC)CNC(C1CC(C(C)(C)O)C1)=O c1(C(=O)NCC(C)CN(C)C(C2CNC(=O)C2)=O)c[nH]nc1C(F)F C1(CCOC)CN(C(=O)CC2(OC)CCC2)CCN1C(=O)CCC1CCCO1 c1(C(N(C2CN(C(C3CC4(CCC4)CO3)=O)C2)C)=O)cc2nc(Cl)ccc2s1 N12CCC(NC(=O)NC)C1C(=O)N(C)C(C)C2=O.c1(SC)cn(C(C)C)nn1 C1(NC(C(C(C)C)SC)=O)CC2(C1)CN(C(c1occc1C)=O)C2 Cc1cc(C(=O)NC2(C)CC(NC(=O)C(C3CCC(=O)N3)C)C2)co1 C1(C)(NC(C(c2ccc(OC)cc2)O)=O)CCCN(C(c2c(Cl)cnn2C)=O)C1 c1(C(=O)NC2C(C)CCN(C(CN(C(C)=O)C)=O)C2)cc(S(N)(=O)=O)co1 Cc1cc2ccc(C(=O)NCCC(C)N(C(=O)CCC3CC3(Cl)Cl)C)cn2c1 C1(CNC(C(CC)SC)=O)CCCC2CN(C(=O)CNC(C3CC3C)=O)CC12 C1(C(N(CCC)CCO)=O)CCCCN(C(=O)C(C)(C)COC2CCCC2)C1 n1(CC)nnc(C(=O)NCC2(NC(C3CCN(C4CC4)C3)=O)CCCCC2)c1C C(=O)(CCCC(C)NC(c1ccc(COC)o1)=O)NC(C)C(C)(C)CN(C)C c1(C(=O)NCCC(C)NC(C2C3(CC(OCC)C3)C2)=O)c[nH]c2c(C)cccc12 N1(C(CCCC#N)=O)CCC2(NC(=O)Cc3ccc4nsnc4c3)CCCC12 C1(NC(c2n(Cc3sccc3)nnn2)c2ccno2)CC2CCCC2C1 CCC(C#N)C(=O)NC1CCCC1NC(c1cc(C(C)(F)F)n[nH]1)=O Cc1ccc(C(C)(CNC(=O)N(C2CC(O)C2)C)CO)cc1 C1(NC(C(C)C(C)O)=O)COC2(C1)CN(C(c1ccc(O)c(F)c1F)=O)C2 c1(CC(=O)NCC2C(NC(CCC(=C)C)=O)CC2)ccc2nc(O)[nH]c2c1 c1(C(N2C(CNC(c3c(C)con3)=O)CCC2)=O)cc(F)c(C)c(N)c1F N1(C(c2nc(C)nc(O)c2)=O)CCC2(CC1)OCCC2NC(C1CCC1(C)C)=O C1(OC)(CNC(=O)NCCC(C)(C)C(=O)OC)CCCC(c2ccccc2)CC1 C1(N(C(C(C2CCCC2)NC(C(C2CCCC2)OC)=O)=O)C)CCN(C)C1 CC1CCC(CC(=O)NCc2cc(C(=O)N(C)CCc3nccs3)co2)O1 C1(NC(Cn2nc(C)c(Cl)c2)=O)CC2CCC1N2C(c1snnc1C)=O N1(C(c2c(CNC(=O)C=CC(=O)NC3CC3)ocn2)=O)CCCCC1CCCO c1(CC)ccc(F)cc1C(=O)N(C)CCNC(=O)C=C1CCN(C)C1 N1(C(C=CC2N(C=CC)CCC2)=O)CC2(CNC(=O)O2)C1.C#Cc1cn(C)nc1CC C1(NC(c2scc(C)n2)=O)CC2CC1N(C(c1cccc(-n3cccn3)c1)=O)C2 C1(CC)C(C(=O)N(C)CC2(CC(C)C)CC2)CCN1C(c1c[nH]c(C#N)c1)=O C(C(C(=O)Nc1ccc(N(C)C)cc1)C(C)C)NC(C1(OC)CCOC1)=O C1(CNC(CN(C(=O)C(C)n2cncn2)CC)=O)CC(CCOC)C1 c1(C(=O)NC(CNC(C(CC#C)C)=O)(C)C2CC2)cnc(O)c2cncn12 CC(CC(=O)NC1CCC12CN(C(c1ccc(Br)o1)=O)C2)C(F)(F)F CC1CCN(C(c2cnc(N)cn2)=O)CC1CC(=O)NCc1cn(C)nc1C(N)=O N1(Cc2cc(OC)ns2)CC(NC(c2occc2Br)=O)CCC1C N1(C(C2C(CCOC)C2)=O)CCC(F)(CNC(=O)C(F)CC2CCCCC2)CC1 Cc1n[nH]c2cnc(C(=O)NCC3COCCN(C(C4(Cl)CC4)=O)C3)cc12 C1(C(=O)NCCc2nc(CO)cs2)COc2cc(F)ccc2O1.CCO c1(C(=O)NC2CCN(C(CCCCOC)=O)CC2F)cc(C)c(C)nc1C C1(CN(C(=O)CC2CC2C)CC)CCN(C(c2cc(C3(C)CC3)on2)=O)CC1 C1(C(N(c2c(C)cccc2)C)=O)CN(C(=O)C(C)(C)C2CCC2)CC12CC2 c1(C(=O)NC2(CNC(C(C)n3cccn3)=O)CCOC2)cc(Cl)ccc1N C1(CC)CN(C(C2CCCCN(C(=O)CC3CCCOCC3)C2)=O)CC(=O)N1 Cc1nc(NCC2CC(CF)C2)cc(O)n1.C12CCC(C1)NC2=O c1(C(N(C2CCCN(C(C3CCNC3=O)=O)CC2)CC)=O)nccc(Cl)c1F C(=O)(CC(CC)C(C)(C)C)N1CCC(NC(C(=Cc2ccc(F)cc2)C)=O)C1C1CC1 c1(NC(CCNC(COC)=O)C)nc2c(cc1C#N)CCC2SC C1(CO)(N)CCCN(CC=O)C1.N1(C(C(=O)NCC2CC2)=O)CC2CCC1C2 c1(C(N2CCC(F)(CNC(Cc3cc(C)sn3)=O)C2)=O)c(F)cc(F)c(F)c1F C1(CC(C)C)CCN(C(=O)C(=O)N(C23CCC2C3)c2ncc[nH]2)CC1 Brc1ccc2nnc(=NCCCN3CCCC3C(F)(F)F)[nH]c2c1 C(C)(CCCNC(c1cc(-c2cccn2C)[nH]n1)=O)NC(C(C)O)=O c1(C(=O)NC2(CC(N3C(C)CC3CO)=O)CC2)ccccc1Cl c1(OCC(=O)NC2CCN(C(C(C)(C)OC)=O)C2)c(Cl)cccc1Cl c1(C(N2CCC3(C(C(N(CCN(C)C)C)=O)C3)C2)=O)ccc(F)cc1C#N C1(NCC2N(C)C(=O)CC2)CC2CCC1(C(=O)NCCN(C)C)C2 C1(NC(CC(C)N(C(=O)C2=CCCC2)C)=O)CCOCC1O c1(C(N2CCN(C(CC3C(CC)C3)=O)CC2CO)=O)cc(N)c(Cl)c(O)c1 Cc1cc(C(=O)NC(C)CCN(C)C(C2CCS(=O)(=O)CC2)=O)n2ncnc2n1 C1(NC(=O)Cc2noc3ccccc23)CN(C(=O)CC(F)F)C2(CCCCC2)C1 C(=O)(C(C(CC)=Cc1ccsc1)N1CCN(C(CC)CC)CC1)NCC=C c1(C(=O)NC(C(C(C)C)NC(CSCCC)=O)C)cc(Cl)ccc1C Cc1cc(Cl)nc(Cl)c1C(=O)NC(C1CCCN(Cc2ccc(Cl)c(F)c2)C1)C c1(C(C(N2CC(N(CC(=O)N(C(C)C3CC3)C)C)C2)=O)O)cnn(C)c1 C1(N(C(C(C2CCCOC2)OC)=O)CC2CC2)CCN(C(=O)C(C)(C)CF)CC1 c1(NCCC(=O)OC(C)C)ccc(S(=O)(=O)NC2CCN(CC(F)F)C2)c(Cl)c1 C1(c2nnnn2C)(NCc2cc(C)n(C)n2)C=CCC(C(C)(C)C)CC1 N1(C(CCSCCCC)=O)CCCC2(CCN(C(=O)CCn3cnnn3)CC2)C1 Cc1nnccc1C(N1CC(NC(=O)C(c2cncnc2)C)C(O)C1)=O C#CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(CC(C)C)COC2)=O)C1 CC1C(C(=O)NCc2ccc3c(c2)CC3)CCCN1C(=O)C(C)NC=O CC1=C(C(=O)N2CCC(F)C(NC(=O)CC3CC(C)(C)CO3)C2)CCCO1 c1(C(N(CCNC(C(C)(C2CCC2)OC)=O)C)=O)nccc2occc12 N1(C(C)=O)CCC(NC(C2(C(c3c[nH]cc3C(C)C)=O)CCCC2)=O)C(CO)C1 C1(NC(CC(CC)C)=O)CCC2(CC1)CC2NC(c1cc(O)nc(C)n1)=O c1(C(=O)NC(CNC(C(N2CCCCC2=O)C)=O)C)cn(C)cc(Br)c1=O C1(NC(c2n(C=C)nnc2)=O)CN(C(c2scc(C)c2Cl)=O)CC1C1CC1 N1(C(=O)NC(c2onc(COC)n2)C)C2CC3C4CC(C3C2O)C4O1 N1(C(CC(C)OCC)=O)CCN(C(=O)CCCCN(C)C(C)C)CC1CO CS(=O)(=O)C1CCC(C(=O)NCC(F)CNC(c2cc(C3CC3)no2)=O)CC1 C1(NC(C(CC)OC)=O)CN(C(=O)C=CCN(C)C2CC2)CC1n1ccnn1 c1(C(=O)NC(C(C)C)(C)CNC(=O)C=Cc2ccnn2C)cccc2ncoc12 N1(C(c2nc(C)sc2C)=O)CCC2CC(CNC(=O)CCCN(C)C)CCC2C1 CC1(C(=O)NCCC(Cc2ccccc2)NC(=O)C=C2CCC2)CCC(=O)NC1 c1(CN2C(C(=O)NC(COC)C)CCC2C)cc(NS(C)(=O)=O)cc(C)c1 N1(OCc2cc(C)c(F)nc2)CCC2CN(C(=O)CC3CCC3)CC12 N1(C(C(C2CC2)OC)=O)CCCC1(C)CNC(c1n[nH]c(=N)s1)=O c1(C(=O)NC2(CCNC(C3(CC)CC3(F)F)=O)CCCC2)ccc2sccc2c1 n1(C(C(=O)N(C(C)CNC(=O)CNC(=O)N(C)C)C)C)cnc(C#N)n1 C1(C2CN(C(=O)CCc3cn(C)nn3)C2)(NC(CC2N(C)CCC2)=O)CC1 CN1CCC(NC(c2cc(CNC(C3CCOCC3)=O)on2)=O)C1(C)C C(=O)(NNc1oc(CC(C)C)nc1C#N)N1C(CC)CCC(C)C1 c1(CC(=O)NCCC2CC(NC(c3cc(C(C)=O)[nH]n3)=O)C2)ncc(F)cc1F c1(C(N(C)C)=O)ccc(CCN(C(=O)CCC2CC2)C2CCSC2)cc1 N1(C(C(P(C)(C)=O)O)=O)CCC2(CCC2)C(CNC(=O)CC2(O)CCCC2)C1 C12(NC(=O)Cc3ccccc3F)CCCC1N(C(=O)COC1CCCC1)CCC2 N1(C(CC2N(C(C3C(C(C)C)CCO3)=O)CC2)=O)CCC(CO)(OC)C1 C#CCC(CC(=O)N1CC(C)(C)CC1C(=O)N(CC(C)C#C)C)OC C(CCCCCNC(C1CC12CC(NC(C1CCOC1(C)C)=O)C2)=O)N(C)C C(C1CCCN1C)=CC(=O)NCCN(C(c1nc(Cl)cs1)=O)CC CCCCS(=O)(=O)N.c1(C(=O)NCC)cn(CCC)nn1.C1C(C)(C2CC2)NC(=O)C1 c1(CNC(C2CC2F)=O)ccc(N)c(C2CC2CNC(C2(CO)CCC2)=O)c1 C(CN=C(NCc1cccs1)NC1COC(C)C1)C1C(C)C1.CC(F)(F)F C1(NC(Cn2c(CCC)ncc2)=O)(CO)CCN(C(c2cc(CC)no2)=O)CC1 O=CC1N(C2CC2)c2ccccc2C1C(=O)Nc1ccc(-c2cnn[nH]2)cc1 CN1C(=O)CCC1C(=O)NC1(CCCNC(=O)CNC(c2ccoc2)=O)CC1 C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(NC(C2(C)CCOC2)=O)C1 c1(C(=O)NCC(=O)NCC(CC)NC(=O)C(C)(C)C)ccc(N)c(F)c1 N1(C(C2CCN(C(C)C)CC2)=O)CC(C)N(C(=O)COC2(C)CCC2)CC1C C(=O)(CC(C)CC(C)C)NCC1N(C(c2cccc(CC)c2)=O)CC(O)C1 CC1(C)COC(CC(=O)NC(CNC(=O)CNS(=O)(=O)C2CC2)C2CC2)CO1 CC1(NC(c2cccn(O)c2=O)=O)CCCN(C(=O)CC2=CCCC2)C1 C(CC(C)C)(C(=O)NC(CNC(=O)C=CC=C(Cl)Cl)CC(C)C)NC(C)=O N1(C(C(CC)NC(N)=O)=O)CCCN(C(=O)CSC2CC2)C(C)C1 N1(C(C(C(=C)C)(C)C)=O)CCc2c(sc(Nc3ncc(C)cn3)c2CO)C1 c1(N(C(CCOCCCNC(C(C)(C)SC)=O)=O)C)cccc(C)c1 Cc1ccc(Cl)c(C(=O)NC23CC(CNC(=O)C4=COCCC4)(C2)C3)c1 C(=O)(C1CCCc2ccccc21)NCCC(C)NC(c1cc(CC(C)C)on1)=O Cc1ccc(CCC(=O)N(CCCC(=O)NC(C)C)C)c(C)c1 CC1(C)C(CNC(=O)CN2CCN(C(c3ccc(O)cn3)=O)CC2)C1(C)C N1(C(COC2CCN(C)CC2)=O)CCC(CO)C(CSc2ccccc2)C1 c1(CC)ccccc1CNC(C1CC(C)CN1C(=O)C(C)(C)C#N)=O C1(CC=C)(NC(c2ccc(C)c(C)n2)=O)CCCN(C(=O)C(N)=O)C1 N1(C(C(=C(C)C2CC2)F)=O)CCOC2CCN(C(C3CCOC(=O)CC3)=O)CC12 c1(C(C(=O)N(CC(O)CNC(=O)Cc2ccccc2)C)N(C)C)ccccc1Cl C#Cc1c[nH]nc1C(=O)NCC1(CC(=O)NCCC(C)C=C)CC1 Cn1ncc(C(=O)NCC2CSCCN2C(=O)CC(=O)OC(C)(C)C)c1C(F)F c1(CC)cc(C)[nH]c(=NCC2CCC(NC(=O)C(C)S(N)(=O)=O)CC2)n1 C1(C(N2CCC(N(C(=O)CC3CCC(C)CC3)CC)C2)=O)CC(=O)NC(=O)N1 N1(C(CN(CCOC)C)=O)CCC(C(=O)NCC#CC#CCO)C12CC2 c1(CC)ccc(C(=O)N(CC(=O)NC(N)=O)CC)o1.c1(CN)nnc(C)o1 N1(C(CS(=O)(=O)NCC)=O)CC(NC(=O)CC(C)O)CC1(c1ccccc1)CSC c1(C(CNC(=O)C(=O)N(C)C)N(C)C)cccc(OC(=O)CN2CCCC2=O)c1 CCC(F)(F)C(=O)NCCCN(C(=O)CC(n1nc(C)cc1C)C)C N1(C(c2cccc(SC)c2)=O)CC(F)(F)CC1C(=O)Nc1ncc(Br)s1 c1(NC(N2CCC(c3ccon3)CC2)=O)ccc(C(=O)C(F)(F)F)cc1 CCCC(CCCNC(=O)C(=CC1CCC(C)CC1)C)NC(C1(OC(C)=O)CC1)=O C=CC(C)(C)CCNC(=O)C(C(C)C)n1cc(-c2ccncc2C)nn1 Cn1ncc2c(N3CCCCC(CNC(=O)C=CC4CCCO4)C3)ncnc12 CC1(C(=O)NC2CCC(n3cc(CCNC=O)nn3)CC2)CCC12CCC2 C(CO)(C(=O)NCc1cc(C(=O)NC2(CF)CCC2)cs1)NC(C)=O C(=O)(C(F)CC(C(=O)OC)NS(=O)(=O)c1ccc(C(C)(C)C)cc1)OCC c1(C(N2CC3OC(=O)NC(C)C3C2)=O)ccc(C#Cc2ccccc2O)cc1 C1(C(N2CC(COC)OCC2)=O)CN(C(c2csc(C)c2)=O)CC12CCC2 c1(Cc2cc(C(N3CC(CC#N)C3)=O)on2)ccccc1Br C(N=c1[nH]c(Cl)ncc1F)C1CCN(C(CC2OCC(C)(C)C2)=O)C1 N1(C(C(COCC)C)=O)CCCCCC1CNC(=O)CCC1CCC1 c1(C(=O)NCC(CN(C(C(C)OCCOCC)=O)C)C)c(N)ccc(F)c1C C1(CNC(C2C(C(=O)OC)C2)=O)CC(C(N2CC(N3CCC3)C2)=O)CO1 n1(CC)nnc(C(=O)NC2(CO)CCN(C(c3coc(CC4CC4)n3)=O)C2)c1C C(=O)(C1CCCc2nccn21)NC1CCN(C(c2ccc(C#N)o2)=O)CC1CO C(=O)(CS(=O)(=O)c1ccccc1Cl)N1C(CNC(C2CCCC(F)C2)=O)COCC1 Cc1oc(C#N)cc1C(N1CCC(O)(CN(C(=O)Cn2ccccc2=O)C)C1)=O c1(CC(=O)NC2(CNC(=O)C=Cc3ncc[nH]3)CCCC2)ccc(Cl)cc1 C1(NC(c2ccnc(C)c2C)=O)CN(C(=O)CC2CCC2)CC(C)(C)C1 C(=O)(CCCN(C)C(c1coc(CNC(=O)C(C2CCOCC2)C)c1)=O)NC C(=O)(C(C(C)(C)C)N(C)C)N1CC(CC=C)(NC(C2CC=CCC2C)=O)C1 Cc1nc2c(CC(=O)OC3CCCCCCC3)cccc2o1 CC1CN=C2NC(C(=O)N3CC(O)(CN(C(=O)CN4CCC(C)C4)C)C3)=NN2C1 n1(CCC(=O)NC2C(NC(C(C)OCC#C)=O)CC2)ccc(O)nc1=O C1(C(N(C)CCC2OCCO2)=O)(NC(C2CCSC2)=O)CC(F)C1 C1(CC(N2CCC(CNCCn3c(C)ncc3)C2)=O)CC2CCC1O2 c1(C(N2CC(OC)C(NC(=O)C=Cc3ccsc3)C2)=O)[nH]nc2ncnc(O)c12 C1(NC(CCCSC)=O)CC(C2CCN(C(c3cc(C)nc4ccnn34)=O)C2)C1 N1(C(C(c2ccc(N)cn2)C)=O)CC2(C)CN(C(C3CC(O)C3)=O)CC2(C)C1 C1(NC(c2ccnc(C(F)F)c2)=O)CN(C(C2(C3CCCO3)CC2)=O)CC1O N1(C(c2scc(OC)c2OC)=O)CC2(CCC(CNC(=O)C3=CCCS3)O2)C1 C1(=CC(=O)N(C2CCN(C(C3CCOCC3OC)=O)C2)CC)CN2CCC1CC2 c1(C(N2CC(O)(C(C)NC(c3cn(C)cn3)=O)C2)=O)ccc(Cl)c(C#N)n1 C(=O)(C1Cc2ccc(Cl)cc21)N(C(c1cn(-c2nccc(C)n2)nn1)C)C CC1CC2(CCO1)CC2C(=O)NCC1C2CN(C(=O)CCCn3cncn3)CC12 c1(C(=O)NC(CNC(C2CCOCC2)=O)C2CC2)ccc2c(c1)COC2=O CC1CCC1N=c1[nH]c2ccc(S(=O)(=O)NC3(C(F)(F)F)CC3)cc2s1 c1(C(N(c2nc(C)cc(OCC)n2)C2CC(N)C2)=O)c(F)cc(C#N)cc1F c1(C(N2C(C)CC(NC(c3c(NCC)scn3)=O)C2)=O)cc(C)cc(Cl)n1 C1(C(N2C(C(=O)NCC(CCC)OCC)C3CC3C2)=O)CC2(CCC2O)C1 Cn1ccc(-n2cnc(C(=O)NC3CCC3NC(=O)CNc3cccnc3)c2)n1 Cc1cc(C)n2ncc(C(=O)NCCC(C)N(C)C(C3COC3)=O)c2n1 C1(NC(C(C=C)(C)CC)=O)CN(c2nnc(C)c(C)n2)CC2(CCOCC2)C1 c1(C(C(=O)N(C)Cc2ccccn2)NC(=O)Cn2cccc2)ccc(F)cc1 C1(C(=O)NCCCNC(c2cc(C(F)F)[nH]n2)=O)CC2CC1CC2O N1(C(CC(CC)OC)=O)CC(C2CN(C(=O)C(CC)CCOC)C2)C1 CC1CNc2c(C(=O)NC(C)CNC(=O)CC3(N4CCCC4)CC3)cnn2C1 C1(C(=O)NCC(C)NC(c2nc(CCC)oc2)=O)Cc2ccccc2O1 N1(C(C(CC)(C)F)=O)CCCCC2(CCN(C(c3cc[nH]c3C)=O)C2)C1 N#Cc1ccc(OCC(N2CC(C(=O)NCC3CCC=CO3)C2)=O)c(Cl)c1 Cc1nc2ncnn2cc1C(=O)NCCCCC1CN(C(c2cnn(C)c2)=O)C1 C(=O)(CCCC(=O)NC1CCCN(C(c2n[nH]cc2Br)=O)C1C)NCC c1(OC)cc(C(=O)NC2CC(C(N3CCCC3)=O)C2)ccc1F.C12CCCN1C2=O C(=O)(N=c1cc2n([nH]1)CCN(CC)C2)N1CCC(C(=O)OCc2ccccc2)CC1 c1(CNC(C2CN(C)C(=O)N2)=O)n[nH]c2c1CN(C(c1sccc1Cl)=O)CC2 n1(CC)ncc(C(=O)N(C(C)CNC(C2(C(F)F)CCCO2)=O)C)n1 C1(CC)CN(C(=O)NC2CCN(c3ccccc3)C2)CC(C)S1(=O)=O c1(COC)nc(C)cc(=NC(C)C2CCCCN2C(c2cc(F)cc(F)c2)=O)[nH]1 N1(C(c2ccc(I)cc2Br)=O)CC2CCN(C(c3cc4ccccn4n3)=O)C2C1 N1(CC(=O)NC2CCCC2C(=O)Nc2ccsc2SCCO)CCC(O)CC1 N(C1CCCc2sc(Cl)cc21)C1CCCN(C(C(=O)Nc2ccc(Cl)cn2)=O)C1 C1(NC(C(C)OCCCC)=O)CCCCN(C(c2nc(C)c(N)cc2C)=O)CC1 N1(C(CC2CCC(NC(C(C)(C)N3CCCCC3)=O)C2)=O)CCC=C(F)C1 C12(C(=O)NCCCNC(C3(C)CC3C(F)(F)F)=O)CC(C(F)(F)F)(C1)C2 C1(C(=O)NCCCN(C(c2c(CCC)occ2)=O)C2CC2)(CC)CCCCO1 C12(NC(C(C(C)C)O)=O)CC(CNC(c3cnn4c3CCCC4)=O)(C1)OC2(C)C C=CCC(C)(CC)C(=O)N1CCC(C(=O)NCC2(C#N)CCC2)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)N1CCC(NC(c2cc(C(C)C)c(N)cc2)=O)C1 CN1CCN(C(C2COCCO2)=O)C(CNC(c2cc3occc3s2)=O)C1 O=C(N=c1[nH]oc2c1CCCCC2)NCC(Cc1cc(Cl)c(F)cc1F)CO N1(CC)CCN(C(c2ccc(OC(F)F)cc2C)C(=O)NC2CCOC2)CC1C C(c1cc(C)no1)=CC(=O)N(CC(=O)NC(C)C(C)F)CCOC CCC(CCC(=O)NCC(CO)NC(c1ccccc1COC)=O)OC C(=O)(C(CC(F)F)C1CCCO1)N1CC2C(NC(C3(C(=O)OCC)CC3)=O)C2C1 C1(C)(C(=O)NCCC2CC(NC(CC(=O)NCC)=O)C2)CCCC1O CCC(O)(CC(=O)N1CCCC(CNC(C2OCC2(C)C)=O)C1)c1ccccc1 c1(C(=O)NC(CN(C(c2cccc(OC)c2F)=O)C)C)coc2c(C)cccc12 N1(C(CN2CC(C)C2)=O)CCC(C2CC2)C1C(=O)NCc1cnc(C2CC2)[nH]1 N1(C(c2c(SCC)cncc2)=O)CCC2(CCC2NC(C2CCCO2)=O)CC1 N#CC1(C(=O)NCC2(CNC(C3(F)CC3)=O)CCCC2)CC=CC1 N1(C(=O)OC)CCCC(N(C(CNC(=O)C=C2CCC2)=O)C)C1 C#Cc1ccc(Cl)c(C(=O)NC2(CNC(=O)C=Cc3sccc3C)CC2)c1 c1(C(N2CCC(CCNC(CNS(CC)(=O)=O)=O)C2)=O)cccc(SC)n1 Cc1oc(C(=O)O)cc1S(=O)(=O)NC(=O)NC12CCC(CO)(CC1)CC2 Cc1cccc2c1OC(C(=O)NC1CC3(NC(=O)C4=CCCCO4)COC1C3)C2 C1(OC)CC(CNC(C2(CO)CCCCC2)=O)N(C(=O)CC2CC3(CC3)C2)C1 c1(C(=O)NCCN(C(=O)COc2ccccc2Cl)CC)cccc2c1COCC2 c1(C(N2C(C)(CNC(C3ON=C(C)C3)=O)CCC2)=O)ncn2cccnc12 c1(C(=O)NC(CN(C(=O)C(C)CC(F)F)CC)C)cc(O)ccc1OC c1(CNc2nccc(-c3ccc(OC)cc3F)c2)ccccc1[N+](=O)[O-] N1(C(C2(Cl)C=CC(C(C)=O)=C2)=O)CCN(C(C2CC2(C)C(C)C)=O)CC1C c1(C(=O)NC2CC(C)N(C(c3ccns3)=O)C2)c(F)cccc1Cl C1(NC(c2c(C)nsc2)=O)CCN(C(=O)C(C)NC(C2CCC2)=O)C1(C)C c1(C(=O)NCCOCCN(C(C(C)OCC)=O)C)cn2cc(C)nc2s1 C1(CC)C(NC(=O)C=Cc2cccc(C)c2)CCCN1C(=O)CCC(C)C C(=O)(CCCCCN=[N+]=[N-])NCC(CNC(C(C(C)C)(C)O)=O)(C)F NC1(Cc2ccc(CCC(=O)N(c3ccccc3)C3CC3)o2)CC(F)(F)C1 N1(C(CC#N)=O)CCC(C(=O)Nc2cc(O)c(F)cc2F)=C(F)C1 C(C)(N(C)N1CCC(C)C1)c1c(C)c(Cl)ccc1.C(C)C CC1CCN(C(c2cc(F)cnc2O)=O)CCN1c1cc(C(F)F)ncn1 C(=O)(C(C)(C)C(C)(C)C)NCC(C)(CC(C)C)NC(c1c(OC)scc1)=O S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1CC(NC(c2ccncn2)=O)CC(C)C1 CN1CCn2ncc(CNCc3nc(C4(F)CCOC4C)n[nH]3)c2C1=O c1(CNC(NC2CC(=O)N(C3CC3)C2)=NCCCCl)cnc2ccnn2c1 N1(C(c2c(CNC(C(C)O)=O)cco2)=O)CC2(C1)CN(C)CCO2 Cc1c(C(=O)N(C)CC2CCCCN2C(c2ncccn2)=O)cccc1Br N1(C(CC(C)(C)C2CC2)=O)CC(CNC(c2cccc(Cl)c2N)=O)CC1(C)C CC(C)(CO)C(CNC(=O)NCCCCc1ccc(Cl)cc1Cl)c1ccccc1 C1(C(N2CCC(CCN(C(CCSC)=O)C)CC2)=O)Cc2ccccc2S1 C=CCCCCCCCC(=O)NC1CS(=O)(=O)CC1NC(C1CCCCC1)=O C(=O)(CC(C)(C)Cc1cn(-c2ccc(Br)c(C)c2)nn1)N(CC(CC)C)C N1(C(CC#N)=O)CCC(F)C(NC(c2ccnc(N3CCCCC3C)c2)=O)C1 Cc1ncc(C(C)NC(=O)COC2CCN(C(=O)CCN3CC(C)C3)C2)s1 Cc1cc(N)cnc1C(=O)N(CCCN(C)C)CCNC(=O)CC1CCCOC1 N1(C(c2cncc(CC)c2)=O)CCN(C(=O)CSC(C)(C)C)CC12CC2 C1(F)(C(N(C(c2ccco2)C)C)=O)CNCC1F C1(C(=O)NC2C(C(=O)OC)CC2)N(C(=O)CCc2ccccn2)CCCC1(C)C c1(C(N(C2CN(C(=O)C(C)(C)c3ncco3)CC2F)C)=O)cc(Cl)cnc1O C1(C(=O)NC2C(CC(=O)NCCC(C(C)C)C)C(O)C2)C2CCC(C2)C1C C1(CNC(CCC(=C)Br)=O)C(C2CC2)CCN1C(c1cnc(C)[nH]c1=N)=O c1(C(=O)Nc2ccc(-c3ccc(COCCC)cc3)nn2)ccc(Br)c(C)c1F n1(CC(=O)NC2(COC)CCN(C(c3c[nH]nc3C)=O)C2)cc(P(C)(C)=O)cn1 C1(NC(COCCC#C)=O)(CC)CCCN(C(=O)CC(C)C(=O)OC)C1 c1(C(=O)Nc2cnn(CCO)c2)cc(-c2ccccc2CCO)cc2[nH]ncc12 Nc1c(C(=O)NC(CNC(c2cc(F)ccc2F)=O)C2CC2)cc(Cl)cc1Cl C(=O)(CCCC(=O)NCCC1CCCN(C(=O)C=CBr)CC1)NCCC c1(CCCCN(C(=O)CC(=O)N2CCCC2)C(C)=O)cn(CCC2CC2)nn1 C1(NC(c2cnc(C)n2C)=O)CCN(C(C2CCN(C(C)C)C2)=O)CC12CCC2 c1(C(C(=O)NC2CC2)N(C)Cc2cncnc2)cnn(C)c1Br c1(CCC(C)(c2nnnn2C(C)C)NCCCCC)ccc(Cl)cc1 C(=O)(C1=NOCC1)NC(C(=O)N(C)Cc1cnsc1)CC1CCCCC1 N1(C(Cn2c(C)c(N)cn2)=O)CCCC2(CCN(C(=O)C(C)S(C)(=O)=O)C2)C1 c1(CC)cccc2[nH]c(C(N3CCC(CNC(=O)C(C)SC)C34CCC4)=O)cc12 C(N=c1[nH]c(-c2ccc(Br)nc2)cs1)c1ncn(C)c1 Cc1ccccc1NC(=O)CNC(=O)NCCC1CCC(F)(F)C1 C1(C(=O)N)CN(C(C23CCC(C2)C3)=O)CCO1.C1(CNC(N)=O)(CO)CCCC1 C12(C(=O)NC(CCC)C3CCC3)CCCC1N(C(C1CCCSC1C)=O)CC2 C1(C(=O)Nc2cccc(NC(C(c3n(C)cnc3)O)=O)c2)CCCC(C)(C)CC1 N12CC3(C1)SCCC3NCCC2=O.CC(C)C(C)COC(F)(F)F.C1(=O)C(F)N1 c1(OCC(N2C(CNC(C=CCOC)=O)C(C)CC2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NCC2(CNC(CC(=C=C)C)=O)CCOCC2)cc(C2CC2)nc(O)c1 C1(C(=O)NC(c2cnn(C)c2)C(=O)N(CCCC)C)CC(C)(C)C1 C(=O)(CC=C(Cl)Cl)NC(C(=O)NCC1(SC)CC1)C C(C(F)(C(=O)NCCc1ncccn1)C(C)C)NC(C(C)(C)NC(=O)OC)=O N1(C(=O)Cc2cccc(Cl)c2)CCC2(CC1)CC2C(N1CCCCCC1)=O CC(CC(F)(F)F)C(=O)NC1CC(CC(=O)N(C2CCC(C)(C)C2)CC2CC2)C1 N1(C(C=COCC)=O)CC2(CC(NC(C3CC3(F)F)=O)C2)C1 C1(NC(CC2(OCC)CCC2)=O)C2CC1N(C(c1cnc(CC)[nH]1)=O)C2 N1(C(C=CC(C)=O)=O)CCC2(CCN(C(=O)C(C)(C)S(=O)(=O)C3CC3)C2)C1 N1(C(c2n(CC)ccn2)=O)CCN(C(C2(C(=O)N(C)C)CC2)=O)CC1C(C)(C)C N1(C(CCCCNC(N)=O)=O)CC2(CCCC2NC(c2ccnc(O)c2)=O)C1 c1(C(=O)NCCCCCN(C(C(C)NC(CC)=O)=O)C)cc(Br)cnc1C c1(C(=O)NC2(C)CC(NC(C3(CCC)CC3)=O)C2)cc2cccnn2c1 C(=O)(CC(C)(C)C(F)F)N1CCC(NC(CSCCC(C)C)=O)(CF)C1 c1(C(C)N(CC(=O)O)Cc2cn(C3CCCNC3=O)nn2)cc2ccccc2s1 c1(OC)c(C)cc(NC(=O)C(C)(C)CN2CCNCC2)cc1C C1(NC(CCc2nnc(C)n2C)=O)CC12CCN(C(C1COC(=O)N1C)=O)CC2 CC1CCCc2c(C(N3CCCCC3CN(C)C(C3(CO)CC3)=O)=O)cnn21 c1(C(C(=O)N2CC(Cn3cc(CCCCCO)nn3)C2)(F)F)ccc(F)cc1Cl c1(C(N2C(C(N(CC=C)CC=C)=O)CC(F)(F)C2)=O)cc2ccccn2n1 C1(CNC(C(C2CCN(C(C3(F)CC=CCC3)=O)CC2)C)=O)CC2CCCC2C1 S(=O)(=O)(c1cc(C(=O)O)cc(Br)c1)NC(CCCC)(C)C N1(C(CCCC(N)=O)=O)CC2CCCC2(NC(c2coc(CC3CC3)n2)=O)C1 C1(NC(c2c(OC)cc(C)s2)=O)CN(C(=O)CSCCOC)C(C)(CO)C1 c1(OC)cc(C(C)Nc2cc(C(=O)O)c(C)c(Br)c2)c(F)cc1F C1(NC(C=CC(C)C)=O)CCCCC1CNC(=O)CCCN1CCCC1 C(=O)(C1CCCn2cc(C)nc21)NCC1C(NC(Cc2cn(CC)nc2)=O)CC1 c1(C(=O)NC2CN(C(c3cnc(CCC)s3)=O)C(C)C2)cc(CC)ccc1N N1(CCC)CCCCC1C(N1CC(=O)CC1C(=O)NCCOCCOC)=O CC1(C)CC(C)(CNC(c2cc(O)nc(Cl)c2)=O)CN1C(=O)COCCF C(C)(C(=O)NCC1CCCCCN1C(=O)CN1CCCC1=O)(C(C)C)OC Cn1[nH]c(CNCC(CO)NC(=O)CC2CNC2)nc1=O c1(C(=O)NC2CCCN(C(c3c(C)noc3)=O)C2)n[nH]c2c1CCSC2 C#CC1CCCN(C(=O)C2=NOC(CNC(C34CCC(CC3F)C4)=O)C2)CC1 c1(C(=O)NC2CN(C(C=COCC)=O)CC2N=[N+]=[N-])c(Cl)nc2ccccn12 N1(C(CONC(c2n(C)c(S)nn2)=O)=O)CC(=O)N2CCCC2C1 N1(C(c2nnc3n2CCC3)C(=O)NC2CC2)CC2(CCCC2)c2c(F)cccc21 C1(C(=O)NC2CCCN(C(CCc3ccc(CC)cc3)=O)C2)CC(C)(C)CN1C c1(C(=O)NC(C(C)NC(C(CCCC)C)=O)C)cc(C)c2ncccc2c1 Cc1cc(C)c(CNCC2CN(C(C3(c4ccccc4)CC3)=O)C2)c(O)n1 c1(C(N(C)CC2CCCN2C(C2(O)CCOC2)=O)=O)cc(C(F)(F)F)nc(Cl)c1 CC1(C(N2CCC(O)C(NC(=O)C=CC(F)F)C2)=O)CCCCCC1 CC1CCCN(C(c2n[nH]c(=N)s2)=O)C1CNC(C1CCNC(=O)C1)=O C(C)(C(CO)NC(C1CCS1(=O)=O)=O)NC(C(C)NC(C)=O)=O c1(NC(CNC(=O)NC)=O)cncc(C(N2CCC(C(=O)OCC)C2)=O)c1 c1(CC)nc(=N)[nH]cc1C(N1CCCC1CNC(=O)CCOCCN(C)C)=O C1(=O)C(C)(C)SCCN1C.S(=O)(=O)(CC)N(CCSCC(=O)OC)C Cc1ccc(O)cc1CNC(=O)CCN(C(=O)C(C)C(C)(C)C)C CCC(CNC(C1(N(C)C)CCCC1)=O)(CC)C(=O)NC1CC(C)OC1=O N1(C(C2(CC)CCCCC2)=O)C(CO)CSCC1c1ccccc1 c1(C(=O)NCC(CNC(C(CC=C)OC)=O)(C)F)cccc(O)c1F C1(C(N2C(CCNC(c3nc(CC)sc3N)=O)CCC2)=O)CCCCC12CCC2 c1(C(C(=O)NCC(=C)C)N(CC(C)CC)CC)ccc(Cl)cc1Br c1(C(N2C(C(C)NC(Cc3nc(C)sc3)=O)CCC2)=O)cnc(C(F)F)c(C)c1 C12(C(=O)NCC(CC)NC(c3ccc(C)s3)=O)CCCCC1C2(F)F c1(C(C(=O)NCCCF)N(CC(C2CCC2)OC)C)ccc(F)c2[nH]ncc12 n1(C(C(=O)NC2(CC(=O)OC)CCC2)C2CC2)cc(-c2c[nH]nc2C(=O)O)nn1 C1(CNC(C(COC)C)=O)CCC12CN(C(c1nc(O)sc1C)=O)C2 c1(CNC2C(C(N(C3CC3)CC)=O)CCC2)cc(Cl)cnc1OC Cc1ncncc1C(N1CC=CC1C(NC[Si](C)(C)C)=O)=O C12(C(=O)NCC(C)N(C)C(c3cnccn3)=O)CC(C(F)F)(C1)C2 C1(C(=O)NCC(=CC(N2CC(=CCC)C2)=O)C)CCCCC1 C(CN=c1nc2sccc2c(NCC2CCC2)[nH]1)(C1CC1)OCC c1(C(=O)Nc2cc(C(F)F)ccc2Br)cc2ccccc2cn1 CCCC(CC)C(=O)N1CCN(C(=O)Cc2cn(C)nc2C)C(c2cn[nH]c2)C1 C1(NC(CC(=C)C)=O)CC(C2CCN(C(c3cc(O)ccc3F)=O)C2)C1 C1(C(=O)NC2C(C=C)COC2)CC2(CC(NC(c3ccn(C(F)F)n3)=O)C2)C1 C(=O)(CS(=O)(=O)Cc1ccccc1Br)NC(C(CC=C)C)=O.C1CC1CN(C)C CC(C)C(O)C(F)(F)C(=O)NCC1CC(O)CN1C(c1ncoc1Br)=O C1(OC)CN(C(c2cccc(CCO)c2)=O)CC1NC(=O)CN(C)C(C)C CN1CCN(CCC(=O)NCC2(C(F)F)CCN(C(c3cnc(O)s3)=O)C2)CC1 N1(C(CSCCOC)=O)CCC(NC(=O)C(F)=C(C)C)C(c2ccccc2)C1 N1(C(CSC)=O)CCC(CF)(NC(c2cc(-n3ccnc3)ccn2)=O)C1 C1(N(C(c2c(C)cc(C)nc2)=O)C)CCN(C(C2C3CCCC23)=O)CC12CC2 C1(C(=O)NCc2c(OC)cccc2)CN(C(=O)CCC2(C)CC2)C(C)(C)C1 C1(NC(C2(C)CC(=C)C2)=O)CC1C1CCCN(C(c2cc3n(n2)CCC3)=O)C1 C1(CNC(c2scc(C)c2)=O)CCCCN(C(c2ccnc(Cl)c2O)=O)C1 C(=O)(CCC(C)C1CC1)NCCN(CCC)C(c1ccccc1-n1ccnn1)=O C1(CC(=O)N(CCNC(c2csc(COC)n2)=O)CC)CCC(=O)N1C C1(CNC(C=CCCCCC)=O)CCC(C)N(C(c2cnsc2)=O)C1 C12(COC)CC(CNC(c3ccccc3SC)=O)(CN1C(c1ccccc1)=O)C2 c1(C(=O)NC2CN(C(C3CC4CCC34)=O)C2)ccccc1N1CCCC1 C1(C#N)(C(=O)NCCCC(C)NC(C(CC)NC(c2ccco2)=O)=O)CC2CC2C1 c1(C(=O)NC(c2cn(CC(=C)C)nn2)C)ccc(SC(C)C)cc1 C(=O)(C1=CS(=O)CCC1)N(C1CCCN(C(=O)CCc2cscn2)C1)CC C1(CNC(c2cc(OC)n[nH]2)=O)CC2CCC1N2C(=O)CCc1ccsc1 Cc1nc2ncc(C(=O)NC3CCN(C(c4cc(F)c(N)c(F)c4)=O)C3)cc2o1 C1(NC(C(C)N(C)C)=O)CN(C(=O)Cn2cccnc2=O)CC12CCCC2 C1(O)(CN(C(C=CC)=O)C)CCCN(C(c2cccc(OCC(F)F)c2)=O)C1 CC1CNCC(CN2CCC(c3ccccc3)(C(F)(F)F)C2)C1 c1(CCC(=O)N(C2CCCN(C(C(CC#C)C)=O)C2)C)ccc(F)cc1F N1(C(CC=C(C)C)=O)CC(N(C(=O)CCC2CC2C)C)C2(CC2)C1 Nc1ccc([N+](=O)[O-])cc1C(N1CC(NC(c2csc(Cl)c2)=O)CC2(CC2)C1)=O C1(C(N2CC(CCn3cc(C4(C)CCCOC4)nn3)C2)=O)CC1C1CCOCC1 N1(C(c2c(C)nsc2)=O)CCCC(C)(C)C1CNC(C1CC12CCCCC2)=O CCCC(CC(C)C)C(=O)NC12CCCN(C(=O)CCNC(=O)OC)CC1C2 CC(C)C(C)(O)C(=O)NC1CCC(CCC(N2C3CCC2CC3)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)NC1CCN(C(C(COC)COC)=O)CC1(C)C Cc1ncc([N+](=O)[O-])n1CC(N1CCC(C(F)CNC(=O)COCCF)CC1)=O C(=O)(C1=CCOCC1)N1C(CCC(=O)NCCCN(C)C2CC2)CCCC1 n1(-c2n(C)ccn2)nc(CCCN(C)C)nc1-c1ccc(C2CC2C)o1 c1(C(=O)NCC(CC)NC(c2ccc(COC)o2)=O)nc(OC)cc(OC)n1 C1(OCCC(=O)OCc2cnc(-c3ccccn3)nc2)CCCCCC1 c1(OCCCCC)ccc(CN2CCC2(C)C(=O)OC2CC2)cc1OC Cc1nn(C)c(-n2cncn2)c1C(=O)NCc1n[nH]c(-c2cccc(F)c2)c1C N1(C(C2N(C(C)C)CCC2)=O)CCN(C(c2c[nH]cc(Cl)c2=O)=O)C(CF)C1 C(=O)(C(C)(C)CCNC(c1ccnc(O)c1)=O)NCC=CC(C)(C)C C(=O)(C(F)C(F)(F)F)NCC(C12CCC(CC1)C2)NC(=O)CCC(F)F c1(OCC)ncnc(OCC)c1C(N1CCC(NC(C2(F)CCCOC2)=O)C1)=O N1(C(=O)NC(CCc2c(C)cc(Br)cc2)C)CCC2(CC1)CN(C)CCO2 N1(C(c2c(OC)ccs2)=O)CCN(C(C2CC(C3CC3)=NO2)=O)C2CCC12 C1(C)(OC)CC(NC(C23CC2CCN3C(c2ccc(OC)o2)=O)=O)C1(C)C c1(C(=O)NC2C(NC(c3cn(C(C)C)nn3)=O)CCC2)ccnc2ccnn12 Cn1cc(C(=O)NCC2(F)CC(CNC(C3CCCN3C3CC3)=O)C2)c(Br)n1 c1(C(=O)NC(c2ccc(Cl)nc2)C)cc(I)ccc1F CN1CCCC(C)(C(N2CC(CCNC(C3CC4(CC4)CO3)=O)C2)=O)C1 N1(C(C=CCN(C)CC)=O)CCOCC1C(=O)N(C1CCCC1C)C C(=O)(C1=CS(=O)(=O)CCC1)NCC1CN(C(C(CCCC)(C)F)=O)CC1(C)C Cc1ccc(C(=O)NCC2CCCN(C(C3CCC(F)(F)C3)=O)C2)cc1 c1(C)cc([N+](=O)[O-])oc1C.c1(NCC)ccn(-c2ccncc2)n1 S(=O)(=O)(c1cccc(N(C)Cc2ccnn2C)n1)NCC(CCC)C Cc1nc(=N)[nH]c(=NCC(C)NC(C2CC(C)(C)OC(C)(C)C2)=O)[nH]1 c1(C(=O)NCC2CN(C(C(=Cc3cccs3)C)=O)C2)cncc(O)c1Cl CC(=O)CCCC(C)C(=O)NC(C(=O)NC(C)C(C)(C)C)C1(C)CC1 C(=O)(C(C)(C)C(=O)NC(C)C(=O)NCc1sc(C)cc1C)OCC Cn1cnn(CC(=O)N(CCC(=O)NCc2ccccc2)C2(C)CC2)c1=O Cc1ccnc(N(C2CCN(C(C34CCC(C)(CC3)OC4)=O)CC2)C)c1[N+](=O)[O-] C1(C(=O)NCCc2c(C(=O)NCC(CC)CC)c[nH]n2)CC12CCOC2 c1(C(=O)NCc2cc(COC)[nH]n2)ccc(CNC(C2CC2C(C)C)=O)s1 C1(C2CCCOC2)(NC(C2C(CNC(=O)C(=O)NC3CC3)CCCC2)=O)CC1 N1(C(C2ON=C(C)C2C)=O)CC2(CCN(C(=O)CN3CCCNS3(=O)=O)C2)C1 C(CC(=O)NN1CCCC1C(N1CCC(CC2CCCS2)C1)=O)=CC c1(C(N2CCN(C(c3c(CCC)onc3C)=O)C3C2C3)=O)cc(C)cc(F)c1N C1(C(=O)OCC)C(F)(F)C12CCC(C(=O)NC1(CO)CCOC1)CC2 CCC(CC(=O)NC(CNC(C1CCC(F)(F)C1)=O)C1CCC1)OC c1(CN2CCC(O)(CNC(CCCCCC)=O)C2)ccnc2ccccc12 C1(C(=O)NC(C)CC2CCN(C(=O)CO)CC2)CN(C)CCN(C)C1 C1(O)(C(C)NC(C(CC)OC2CCCC2)=O)CCN(C(C2OCC2(C)C)=O)CC1 c1(CC(=O)N(CC(CNC(Cn2ncc(CC)c2)=O)(C)C)C)cnccc1OC N1(c2ncc(C)cn2)CCCC1C1CCCCN1C(c1cccn2ncnc12)=O c1(C(=O)N(c2cnccn2)C2COC2)cccc2c1OCCO2 C=CC(CCC)CC(=O)N(C(C)C(=O)NC1COCC(C)(C)C1)C1CC1 N1(C(c2cn(C3C(OCC)COC3)nn2)=O)CC(C(=O)OC)C2(CC2)C1.CC(=O)OC c1(C(=O)NC(CCNC(C2C(C)CN(C)C2)=O)(C)C)cc2nccnc2cc1F C1(NC(C(=O)NC2CC2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C12CCCC2 C(c1ccc(Cl)cc1)=CC(=O)NC12CCN(C(=O)Cc3c[nH]nc3O)CC1C2 C1(NC(CCC2C(C)(C)C2)=O)CCSC12CN(C(=O)Cc1cc[nH]c(=N)c1)C2 c1(C(=O)NC(C2CN(C(=O)CC3(O)CCCC3)CCO2)C)cc2cccnc2[nH]1 C(N=c1[nH]c(=NC(C)c2csc(C)n2)c2c(ncn2C)[nH]1)C1C(C=C)C1 N1(C(c2c(CC)ocn2)=O)CC2CC1CC2NC(c1cc(Br)cn1CC)=O N1(C(c2cc(OC)n(C)n2)=O)CCC(C)N(C(C2CCCCC(C)(C)C2)=O)CC1 c1(C(=O)OC)cc2cc(N(C)Cc3c(N)cccc3Br)ccc2o1 C1(CCOC)(NC(c2ccn(CCC)n2)=O)CC(F)(F)C1 C(=O)(NNc1cc(C)nc(-c2ccccn2)n1)CC(=C)C c1(OC)cc(C(=O)NC2CC(CCNC(C3(C)CCC3)=O)C2)ccc1O c1(C(N2CC(CNC(c3nnc(C)s3)=O)N(C)CC2)=O)ccc(S(N)(=O)=O)s1 N1(C(C2(COCC#C)CC2)=O)CCC(C(=O)NCCCC(=O)O)C(C)(C)C1.C1(CCC)CC1 c1(C(N2CC(C)C(NC(c3cccc(Cl)c3)=O)C2)=O)cc2cc(F)ccc2o1 c1(OCC)cccc(CC(=O)NCC2CN(C(=O)Cc3cnsc3)C2)c1[N+](=O)[O-] Cc1cccc(CCC(=O)OCc2cn(C)nc2O)c1 N1(C(C2CCC(N(C)C)CC2)=O)CCCC(NC(C2(O)CC(C)(C)C2)=O)C(F)C1 N1(C(C(CCC)C(C)C)=O)CCC(N=c2[nH]c3cc(Br)cnc3s2)CC1 Cc1ccc(C(N2CC3(C)CC2(C(N2CCC(O)(C(C)C)C2)=O)C3)=O)cc1F C1(O)(CNC(c2ccn(C(F)F)n2)=O)CCN(C(=O)CCOCC2CCC2)C1 O=C1CN(C(=O)CNC(=O)CC(O)C2CC2)CC2(CC2)N1 c1(C(N2C(CNC(C(C=CC)O)=O)CCCC2)=O)c(Cl)cccc1C#N c12cn(nn1)CC2.N1(CC(=O)NCC(=O)N(C)C)CCOC1=O.C1CS1 C=CCCC(F)(F)C(=O)NCc1ncoc1CCNC(C1CCCS1)=O CC(O)CCCCCC(=O)N1CCC2(CC1)CC2NC(c1c(C(F)F)cnn1C)=O C(C(=O)N=c1ccn(CCF)[nH]1)COC1(C)CCOCC1.C1C(=O)N1 c1(CC)ccc(C(=O)NC2CC(CCNC(C3CCS(=O)CC3)=O)C2)c(F)c1 C(C(F)F)(C(C)(C)C)NC(CC(C)(C)N(C(c1cncc(OC)c1)=O)C)=O c1(C(N2CC3C(CNC(c4c(C)cc[nH]4)=O)(C3)C2)=O)cnc2ccnn2c1C c1(-c2cn(C(C)CNC(c3cc(Cl)c(Br)s3)=O)nn2)cnccc1C#N C(CC(=O)NCCCC1CCC1)(C(F)(F)F)NC(C(C)N(C(C)=O)C)=O Cc1ccc(SCC(=O)NC2(C)CCN(C(C3C4CCC34)=O)CC2)cc1C Cc1cccc(C)c1CC(N1CC2CC(NC(=O)Cc3nocc3C)C1C2)=O C1(NC(NCC2(c3c(C)cccc3C)CC2)=NCCCCl)CCc2ccccc2C1 C(N=c1[nH]c(=NCC(C)(C)OC)c2ncccc2[nH]1)C1C(C=C)OCC1 C1(C(N(C2CCN(C(=O)Cc3conc3C)CC2)CC)=O)CCn2nnnc2C1 N1(C(C(C2CC2)OCC)=O)CCS(=O)(=O)C(CCNC(c2c[nH]c(=O)cn2)=O)C1 C=CC1CN(C(=O)C(CNC(c2c[nH]c(=NC)o2)=O)CC2CC2)CCO1 C1(CNC(C(=O)NCC)=O)CN(C(c2ccc(C(F)F)o2)=O)CC1O c1(C(N(C(C)C(N2CCC(SC)CC2)=O)CC)=O)ccc2cncn2c1 C1(CC(=O)N(C(C)C(=O)O)CCO)CCN(C(=O)C(c2ccccc2)C)CC1 S(=O)(=O)(c1cccc2c(Cl)nccc12)N1CC2CN(C(C3CCC=CO3)=O)CC21 C=C(F)C1(CC(=O)NCC(C2CC2)NC(C2(CCOC)CC2)=O)CCC1 N1(C(CCC2CC(OC)C2)=O)CC(CNC(=O)Cc2conc2C)C(C)(C)C1 C(=O)(C#CC1CCOCC1)NCC(C(C)C)(C)NC(=O)CCc1ccc(O)nn1 CCCCC(C(=O)NC(C)CNC(=O)Cc1ccns1)C(C)C C(C)(C)(C(=O)NCC1CCCN1C(=O)C(C)c1ccsn1)SC c1(C(=O)NCCCO)ccccc1-n1cc(Nc2nc(O)cs2)nn1 C12(NC(CC(C)OC)=O)CCCC(CN(C(C3(CF)CCOCC3)=O)C1)C2 N1(C(c2c(CC)ocn2)=O)CCN(C(C2CC=CC2)=O)CC1C(C)(C)C Cc1cc(C(C2CC2)NC(C2C=CCN2C(C23CCCC2CCC3)=O)=O)cnc1C C1(NC(CCc2cn(C)nc2)=O)CCN(c2ncc(I)cn2)CC1O c1(C(=O)NCC2C(CNC(c3cc(OC)nn3C)=O)C2)nccn2ccnc12 C1(CNC(c2cc(OCC)n[nH]2)=O)C(C)CCCN1C(c1cocc1C)=O C=CCC(Cc1ccccc1)C(=O)NC(C)C(CO)NC(=O)Cc1sccc1C N1(c2n(CCC#C)c(-c3ccc(OC)o3)nn2)CCN(C)C(C)C1C N1(CCNC(C2C3CCC23c2ccccc2)=O)CCN(C(c2ccoc2)=O)CC1 Cc1cc(C)c(C(=O)NC2CN(C(=O)Cc3cnn(C)c3)CC3(CC3)C2)c(O)n1 C1(CSCC)CCCC1NC(=O)Nc1ncc(C(=O)OC(C)C)o1 C12(NC(c3ccc(C)n3C)=O)CCN(C(c3ccc(C(N)=O)cc3)=O)CCC1C2 C(=O)(CCC1=CCc2ccccc21)NCC(CCNC(C=CS(C)=O)=O)O N1(C(c2c(COC)cccn2)=O)CC2CCC(C1)C(NC(=O)C(C)CC1CC1)C2 c1(C(N2CCN(C)CC2CNC(C2(C)CC(F)C2)=O)=O)ccc2c(c1)COC2=O C(C(C(C)C(C)C)NC(=O)Cc1ncn(C)c1C)NC(c1c(CCC)n[nH]c1)=O c1(-c2n(Cc3ccc(C)cc3)nc(C3CC34CC4)n2)cc2c(Br)cc(F)cc2[nH]1 c1(CC)ccc(C(N2CCC23CN(C(=O)C(C)(C)C(C)C)C3)=O)cc1C#N c1(C(N2C(C)CC(NC(C3COCCOC3)=O)CC2)=O)cnn2c(=O)cc[nH]c12 CC(CNC(C1CC1C1CC1)=O)CC(=O)NOCCc1ccccc1 CC(C)(CC(=O)N1CCC(C)(CCNC(c2coc(C(F)F)n2)=O)C1)C(F)F Cc1nc(O)sc1C(=O)NC(c1cn(C)nn1)C(=O)NCCOC1CCC1 C(=O)(C#CC1CCCCC1)NCC(C1CCOC1)NC(c1c(CC)nc(C)s1)=O c1(CN2CCN(C3CCN(C(CSCC)=O)CC3)C(=O)C2)cccc2sccc12 C(=O)(C(C#N)C(C)(C)C)NC1COCC1CN(C)C.c1(COC)cc[nH]c1C=O c1(C(=O)NC2C(NC(COc3cn(C)nc3)=O)CCOC2)c(Cl)ccc2c[nH]nc12 c1(CC)nc(C(=O)NC2CCCC(CNC(=O)C(C)(C)OC)C2)c(N)s1 C1(C(=O)NC(c2ccnc(C)n2)C)COCCN(CCOCC(C)(C)O)C1 c1(OC)ccccc1S(=O)(=O)N1CC2(CCN2C(=O)CSC(C)C)C1 C(=O)(CC(CC)CCC)NCC(CCCC)NC(=O)Cc1ccc2c(c1)CCC2 C12(C(N(C)Cc3c(C)noc3C)=O)CC(CO)(CN1C(C1CC(=O)CS1)=O)C2 CCCCCC(=O)NCC(CC(C)C)NC(C1(C(N)=O)CCC1)=O C(CC(C)C)(C(=O)NC1CN(C(C2COCCN2C)=O)CC1C)OC c1(C(N2CCC(C(N3CCC(CCN)C3)=O)CC2)C)ccc(F)cc1F n1(CCC(=O)N(C2CCN(c3nccc(CO)n3)C2)CCC)ccccc1=O C(=O)(CCCC(=O)N1CCC(O)(CCNC(c2c(Cl)csc2Cl)=O)C1)OC CC1(C)C2CCC(NC(=O)CCCNC(C34CCCC3C4(F)F)=O)C1C2 c1(OC)cc(Cl)ccc1NC(c1cccc(C(N)=O)n1)c1nnnn1C(C)CC c1(C(=O)NCCOCCNC(C2(C)CCOC2)=O)cc(Cl)c2c(c1)OCCO2 c1(C2C3CC(C)(C3)N2)ccccc1Cc1cc(C(C)(C)C)ns1.CC C1(CCCCCNC(C(C=C)O)=O)CCN(C(=O)CCCC=C)CC1 CC1=C(C(=O)NCC2(NC(C3CC3Cl)=O)CCCCC2C)CCS1(=O)=O N1(C(COCc2cc(C)on2)=O)CCCN(C(=O)CC2CC2)C(C(C)C)C1 C1(NC(CCNC(CSCCCC)=O)=O)CC(O)C(O)C1 C(=O)(C(F)CC(C)(C)NC(c1cn(C)cn1)=O)NCC(C(=O)OC)(F)F c1(OCC)cnc(C(=O)NCC2CCC(NC(=O)C(C)(Cl)Cl)C2)cn1 N1(CC(=O)Nc2ccccc2)CCC2(C1)OCC1CC21.C12COCC1C(=O)N2 CC(C)(O)C(F)(F)C(=O)NCC1(O)CN(C(=O)CCC2CCCOC2)C1 N1(C(C2(CSC)CCC2)=O)CC2CC(C1)N(C(=O)Cc1c[nH]nc1C)C2 c1(OC(C)C)ccc(C2CCN(C(=O)C(=O)NC(CC(Cl)(Cl)Cl)C)CC2)cc1 N1(C(C(=O)N(CCC)CCNC(=O)CC(C)n2ccc(C)n2)C)CCCCC1=O C12CCN(S(=O)(=O)N3CCC(CC3)C(=O)NC1COC)CC2.C(C)(=O)OC CC(C)(C#N)CCC(=O)N1CCCC1C(C)(C)NC(C1(C)CCN(C(C)=O)C1)=O C(CN=C(NCC1CCC(CC)CC1)NCC(C)(C)C)c1ccc(SC)cc1 CC#CCCCCN=c1cc(C)c(S(=O)(=O)N2CC(NC(=O)CC)C(C)C2)c[nH]1 c1(OCC(=C)C)ccccc1CC(=O)NCCC(C)NC(c1ccnn1CC)=O C1(CC(=O)NC2CCSC2)CCN(C(=O)N(c2ccccc2)CCCl)C1 Cc1cc(C(N2CCC(N(C(=O)C(N3CCCC(O)C3)C)CCO)C2)=O)n(C)n1 c1(NC2(C)CCCN2C(c2ccc(C(=O)OCC)[nH]2)=O)cnccc1OC c1(NC(C2(NC(CC=C)=O)CC2)=O)cc(Cl)cc(Cl)c1Cl CC1C(C)N(C(=O)C(CN(C)C)N(C)C)CCN1C(C1(C)CCN(C)C1=O)=O Cc1nc2cncc(C(=O)NCC34CC3CN(C(c3ccns3)=O)C4)c2[nH]1 CN1CCOC(C(=O)NCc2ncoc2CNC(=O)CCc2nccn2C)C1 C1(CC=C)(NC(=O)CCOC2CCCOC2)CCN(C(=O)C=CC(=O)NC2CC2)C1 C#CC1(C(=O)NC2CC=CCC2C)CN(C(=O)Cc2ccccc2F)C1 C(C)(C)(CCCNC(=O)C=Cc1cn[nH]c1)NC(C12CC(OC)C1C2)=O c1(C(F)F)nc(=NCC2CNCc3ccccc32)c2c([nH]1)CCCC2 N1(C(C2(C)N(C(c3ncc(C)cc3C)=O)CCC2)=O)CCC2=C(CCCC2)C1 C1(C(=O)NC(C)CNC(=O)C(C)(C)CN2CCN(C)CC2)C(C)(C)OC1(C)C Cc1c(N(C(C)CN2CCOCC2)C2CC2)nc[nH]c1=NCC1C=CCC1 CC1(C)COC(CCNC(C2CC(N)C2(C)C)=O)C1 c1(OC)cc(N2CC3(CCC(C(=O)NC(CO)CO)CC3)C2)nc(S(C)(=O)=O)n1 C(CCCCCCC)CN1CCC(O)(CC(=O)N(C(C(C)=CC)=O)CC(C)C)C1 C(CC(C(=O)NCC1CCC(=O)O1)NC(C)=O)SC C1(C2(O)CCOCC2)(C(=O)NCC2(F)CCN(C(c3cnc(C)[nH]3)=O)C2)CC1 C(=O)(CC(O)CCSC)N1CC(CCCNC(CC)=O)OCC1 N1(C(CC(=C)C)=O)CC2(CCC(NC(C3(C)CC3C(F)(F)F)=O)CC2)C1 C1(F)(C(=O)NC(CSCC)CO)CCN(C(=O)CC2CCCC3CC23)C1 Cc1c(C(=O)NC2CN(C(c3ccncn3)=O)CC2C)sc2cncn12 N1(C(Cc2nnc(C)o2)=O)CCC(C)C1CNC(c1scnc1C(F)F)=O c1(C(N(CC(C)CC(=O)OC)CC)=O)c(C)cccc1C N1(C(C2CC(F)(CO)C2)=O)CCCOC(CNC(C2(O)CC2)=O)C1 N1(C(CC2OCC(=O)C2)=O)CCCC(C2CCN(C(C34CC5CC3C4C5)=O)CC2)C1 c1(C(C)C)cnc(Cl)[nH]c1=NC(C)C1CC(=O)N(c2ccccc2)C1=O C(=O)(C(F)(CC)C(=O)OC)NCCC(CC)(CC)NC(C(C)OCC#C)=O CC1CCc2[nH]nc(C(=O)NCCCC(C)NC(=O)CCc3ccccc3)c2C1 N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CCN(C(=O)Cn1ncnn1)C2 Nc1cc(C(N2CCCC(NC(c3ccnc(Cl)n3)=O)CC2)=O)cc(O)c1Cl N1(C(c2c(CC)cncc2)=O)CCC(C(=O)NCCN2CCCC(O)C2)C12CC2 C1(Nc2nc(C)cc(C)n2)CCCC12CN(C(c1cnn(C)c1C)=O)C2 C1(CC)C(NC(c2sc(OC)nc2Cl)=O)CCN1C(=O)C=Cc1ccccn1 c1(NC(C)C)nc2ccc(C(N3CC(C)C(F)(F)C3)=O)cc2s1 CC1CC(C(=O)Nc2nnc(-c3cccnc3)s2)=NO1.C12CC(F)(C1)CNC2=O N1(C(c2cccc(C)n2)=O)CCC(NC(=O)C(C)NC(C2CCCC2)=O)CC1C C1(OC)CC(C)CN(C(c2c(C)noc2C)C(=O)NCCC2(C)CC2)C1 CCCCCCC(C)n1nc(-c2ccc(OC)cc2)nc1Cc1c(C)nn(C)c1C C(C(C)(C)C(C)(C)C)NC(C(CC=CC)NC(c1cccc(F)c1F)=O)=O c1(NC(CSCCNC(Cc2ccc(C)o2)=O)=O)cccc(Cl)c1C Cc1cccc(N)c1C(=O)NC1CCC(N(C(=O)C2=CC(C)(C)C2)C)C1 c1(NC(=O)CCC2(C)CN(C(CN3CCC(C)CC3)=O)C2)c[nH]c2ccncc12 c1(C(=O)NCc2cn(C3C=CCCC3)nn2)ccc(C(=O)O)c(C(F)(F)F)c1 N1(C(c2cc(C3CCOC3)[nH]n2)=O)CCC2(CCCN2C(=O)Cc2nc[nH]n2)C1 c1(C(N2CCC(N(C(c3cc(C)on3)=O)C)C2)=O)ccc(C2CC2)nn1 CC(CCC(=O)NOCCCCF)NC(C1CC12CCC2)=O c1(C(=O)NCCC(C)NC(C2CC2C(F)(F)F)=O)csc(-c2ncc[nH]2)n1 c1(C(=O)NCCCC)cnn2cc(-c3sccc3CO)ccc12 CS(=O)(=O)c1ccc(F)c(C(=O)OC2CCC3(CCOCC3)C2)c1 C(=O)(N1CC2COCC2O1)C1C2N(C(c3nccc(CC)c3)=O)C(CC2)C1 CCCCCCC(CC)C(=O)N1CCC(O)(CNC(C2CN(CC)CCO2)=O)C1 C1(C(=O)NCC(CCOC)O)CCN(C(=O)c2csnn2)O1 CC(C)C1=NOC(C)(C(=O)OCc2cscn2)C1 C12(CCNC(=O)C(c3cc(F)cc(F)c3)O)CCC(CC1)N(C(=O)CSC1CC1)C2 C1(NC(c2c(C)con2)=O)CCCC(NC(=O)CCCCN(C)C(C)C)C1 N1(C(c2c(C)occ2)=O)CC2(CC(CNC(C3CC3c3cnnn3C)=O)C2)C1 C(=O)(C(C)S(N)(=O)=O)N1CCC(C(=O)NC(CC)C(C)(F)F)C1 C1(SCC(=O)N(C2CC(NC(=O)CN3CCN(C)CC3)C2)C)CC2(CCC2)C1 Cn1c([N+](=O)[O-])cnc1C(=O)NCC(F)CNC(c1cccc(N)c1C(F)F)=O c1(C(=O)NCC2CC(NC(C3CC(C)SCC3)=O)C2)cc2c(=O)[nH]ccn2n1 C(C(C)(C)CNC(C1CC1C#N)=O)N(C(=O)C(=O)NCC(F)F)CC c1(N(C2CC(NC(=O)CCc3ccc[nH]3)C2)C)ccc(C2CCCO2)nn1 C1(O)(C(C)NC(c2c(C(C)=O)ccs2)=O)CCN(C(=O)Cn2cnnc2)C1 C1(NC(c2cc(C(F)F)[nH]n2)=O)CC(F)(CNC(C2CCS2(=O)=O)=O)C1 CN1CCCC(Cc2nc(-c3cccc(F)c3)nn2CCS(C)(=O)=O)C1=O C1(CC)(NC(=O)Cc2cnn(CC)c2)CCCN(C(=O)CSc2ccncc2)C1 N1(C(C(C)N2CCC2)=O)CCC2(CC1)CN(C(c1c(C3CC3)cnn1C)=O)C2 c1(C(=O)NCCC2CN(C(C(c3ccc(F)cc3)OC)=O)C2)cc2ccsc2s1 c1(OCC(CN2CC(CC)C(O)C2)O)cccc(C)c1C C1(C2CCCN(C(c3cccc(F)c3SC)=O)C2)(NC(C(C=C)O)=O)CC1 n1(CC)nccc1C=CC(=O)NC12CC(NC(C3C4CNC(=O)C34)=O)(C1)C2 c1(OC)cncc(C(=O)NC(C2CCCN2C(c2csc(C(N)=O)n2)=O)(C)C)c1 C1(NC(c2cc(=O)cc[nH]2)=O)CN(C(c2ccn(CCO)c(=O)c2)=O)CC12CC2 N1(C(c2ncn(CC)n2)=O)CCCC(C2CCN(C(c3ccco3)=O)CC2)CC1 c1(C(N(C2CN(C(=O)C(F)(F)CO)CC23CC3)C)=O)ccc(C2CC2)nc1O C1(NC(C2CC(SC)C2)=O)CN(C(c2[nH]ccc2C)=O)C(C)(C)C1 C1(C(=O)NCCCN(C(=O)CN2CCN(C3CC3)C2=O)CC)CC12CC(O)C2 c1(C(N2CCC(N(C(c3cc(CC)on3)=O)C)C2)=O)cc(=O)cc(Cl)[nH]1 CC(C)C(C(C)NC(=O)CCC(=O)N1CCCC1)NC(=O)C(=O)NCC(F)F Cc1c(NC(C2CN(C(C3CC(C)(C)CCO3)=O)CCN2C)=O)cccc1F N1(C(C(CC#C)C2CC2)=O)CC=C(C(C)(C)C(=O)NC2(C)CCCC2C)C1 CC1CCN(C(C2CCCC(O)C2)=O)CCN1C(c1ccno1)=O N1(C(c2nccc(N)c2Cl)=O)CC(CNC(=O)Cc2ccoc2)N2CCC1C2 C#Cc1c[nH]nc1C(N1CCC(F)(C(=O)NC2(C)CCOC2=O)C1)=O N1(C(C2CCOCC2)=O)CCC2(CC1)CC2(CO)CNC(C1(O)COC1)=O c1(CN2CCN(C(c3ccncc3)=O)CC2)ccc(O)c(F)c1F N1(C(C(CC(C)C)C)=O)CC(NC(=O)CCCOC(C)(C)C)CC2(CC2)C1 C(=O)(C1CCCc2nc[nH]c21)NC1CN(C(Cc2c(C)ccnc2)=O)C1 CCCCC(O)CCC(=O)NCC1CC2COCC2N1C(c1cnc(Cl)[nH]1)=O c1(C(=O)NC2(CN(C(CC(CC)C(F)F)=O)C)CC2)ccc2cccc(Cl)c2n1 N1(C(C(N2CCCC(O)(CCOC)C2)=O)=O)CCOC2(CCN(C)C2)C1 C(=O)(C(C)(F)C(=O)NCC(O)CNC(c1n[nH]cc1Br)=O)OC N1(C(CN(C)C)=O)CCOC(C(N2CC(N(C)C)C(F)C2)=O)CC1 C(=O)(C1=C(C)CCOC1)NCC1N(C(Cc2ccc(OCC)cc2)=O)CCCC1 N1(C(C)CNC(c2ccc(CO)o2)=O)CCN(C(=O)CCN2CCCCC2)CC1 N1(C(C2CN(C(CC)C)C(=O)C2)=O)CCOCC(NC(c2cncnc2)=O)C1 Cc1ccc2c(=NCCOc3ncccn3)[nH]c(N3CCC(C#N)C3)nc2c1 N1(C(c2nc(CCCC)oc2)=O)CC2CCN(C(=O)CC3CC(C)=NO3)C2C1 N1(C(c2cc(C)n(C)n2)=O)CC2(CCC2)CC1C(=O)N(C)OCc1ccccc1 C1(CNC(C(=O)Nc2c(C)n(C)nc2)=O)CCc2cncn2C1 c1(OC)ccc(CC(=O)N(C2CCN(C(=O)CC(=O)OC(C)=O)CC2)C)c(C)c1 C12CCCCN1C2=O.CC(C)(C)N(CC=CC(=O)NC1COC1)C1CC1 C(=O)(CCCC(F)(F)CO)N1CCCC(CN(C(C2CC2(F)F)=O)C2CC2)C1 Cn1nnc2c1C(C(=O)N1CC(NC(c3ccnc4c3ncn4C)=O)C1)CCC2 Cc1cc(CC(=O)NC2(C(=O)NC(C)CN3CCCC3=O)CC2(C)C)cc(C)c1 c1(N(CC(N2CCCC2C2(O)COC2)=O)CC)cccc(C)n1 C(=O)(CCC1CCc2ccccc21)NC1(N(c2nc(-n3cccn3)cc(C)n2)C)CC1 C(=O)(CC(C)(C)C(C)(F)F)N(C1CCN(C(CS(CC)=O)=O)C1c1ccccc1)CC c1(CC)cc(C(=O)NCC2CCCCC2NC(=O)CN(CC(C)(C)C)C)nn1C N1(C(c2c(OC)cccn2)=O)CCCc2ccc(NC(C3CCCO3)=O)cc21 c1(-c2cn(C)nn2)nnc(CCC2CCCO2)n1CCC#N N1(C(=O)NC(C)C)CCCC1C(=O)NCC1CN(C)C1.C12CCN1C2=O c1(CNC(c2nnnn2C)CCOCC)ccc(OC2CCCC2)cc1C C1(NC(C(CC#C)C2CCCCC2)=O)CCCN(C(c2cnnc(C)c2)=O)C1C C(=O)(C(CC(F)F)NC(C1CCC(F)(F)C1)=O)N(C)Cc1c(C)ncs1 C1(C(=O)OCC)CCC(=O)C(NC(=O)CC2(OC)CCC2)C1 N1(C(CCOCC#C)=O)CCCCC1CN(C(=O)C=C(Cl)Cl)C O=C1CS(=O)(=O)CC(C(=O)NC2(CNC(=O)COCCOCCO)CCOC2)N1 C(CNC(c1cncnc1C)=O)(CC)(CC)NC(c1c(CC)noc1)=O C1(CNC(=NC)NC2CCN(CCc3ncn(C)n3)CC2)CC(=O)N(C)C1=O Cc1ccc(C(N2CCN(C(=O)CCc3cncs3)CC2CF)=O)c(N)c1Cl N1(CC)CCCC1C(=O)NCCCC(C)NC(C1(C(=O)OC)CC1)=O c1(C(C)=O)cc(NC(C2(O)CN(C(=O)COCC(N3CCCC3)C)C2)C)ncn1 C1(C(=O)NCCCN(C(C(C(C)C)OCC)=O)C2CC2)CCCCC1(F)F N1(C(C(=O)NCC)C(C)=C(C)C)CC(NC(c2cc(C)nc(C)n2)=O)CCC1C c1(CC(N2CC(CC(C(=O)OC)F)C2)=O)ccc(C(C)=O)cc1 C(=O)(C(C)CC(C)(F)F)NCCc1ccc(CNC(C(CC(=O)OC)C)=O)cc1 C1(C(=O)NC2(c3c(OC)cccc3)CC2)CCCCN(C(C2CCN2C)=O)C1 c1(C(=O)NCC2C(CNC(COCC(=O)NC)=O)C2)nc(C)ncc1Br C(CCCCCCO)N(C(C(CC)C)C)CC(=O)OC(C)C N1(C(CC)=O)CC2(CCCN2C(=O)C(CC)CCNC(=O)OC(C)(C)C)C1 C#CC1(O)CCN(C(c2noc3c2COCC3)C(=O)NCc2ccco2)CC1 C1(C(=O)NCC(C)C2CC2)CN(C(c2cnn(C)c2)=O)CCO1 C1(C(=O)O)(NC(C(CC)n2ccnc2)=O)CCC(Cn2cccn2)CC1 C1(C(N)=O)CN(C(C2CSCCN2C(=O)Cc2ccc(O)cn2)=O)CC12CC2 C1(CNC(c2c(C(C)C)noc2)=O)CCCC(NC(=O)C(F)C2CCC2)C1 C1(CC=C)(NC(=O)Cc2cnnn2C)CCN(C(c2ccc(SC)s2)=O)C1 c1(NCC2N(C(c3n4cc(C)sc4nc3)=O)CC2)ncnc2c(Br)cccc12 c1(OC)cc(CNC(C2CC2C(=O)Nc2ccc(Cl)cc2Br)=O)cc(C(C)C)c1 C(=O)(CCC(C)NC(=O)CN(C(=O)C(C)C)C)NCC1(CC)CCCC1 C#CCC(CC#C)C(=O)N(C)CCOCCCNC(=O)CC(C)SC N1(C(C(C)Oc2ccccc2)=O)CCC(O)(CNC(C2(C)CCNC2=O)=O)CC1 C(=O)(C(C)(C)CNC(C)=O)NCCCCCNC(C1C(=C)C1)=O C1(NC(CC2(C)N(C(c3cncn(C)c3=O)=O)CC2)=O)C2CCCC1COC2 c1(C(c2nnnn2CCC2CC2)NC(CCSC)C)c(C)cc(N(C)C)cc1C CCCC(O)CC(=O)NC1C2CC1CN(C(=O)CCc1c(F)cccc1Cl)C2 N1(C(C(CSC)C)=O)CCC(c2cc(CNC(C3CCCCO3)=O)on2)CC1 C(=O)(N=c1cc(C)n(-c2ccc(Cl)cc2)[nH]1)C1C(NCc2nnc(C(C)C)s2)CC1 c1(C(C(=O)NC2CCN(C(C(CC)=CC)=O)C(C)C2)(F)F)ccc([N+](=O)[O-])cc1 N1(C(CCc2ccc(C(C)=O)s2)=O)CC(NC(=O)C(C)O)CC2(CCC2)C1 C1(NC(CC=C(C)C)=O)CCCCN(C(c2cnc(OC)c(C(F)(F)F)c2)=O)C1 C1(NC(C(COCc2ccccc2)N(C)C)=O)CCN(CCO)CC1 Cc1c(C(=O)NC2CCC(CNC(=O)C(F)=C3CCC3)C2)sc2cncn12 c1(NC(c2[nH][nH]c(=N)c2C#N)C)[nH]c(=NCC2CCC(C(N)=O)C2)nc2sccc12 C1(CC(=O)NCc2ccc(C(N(C(C)C(C)C)CC)=O)o2)CC(C)(C)CO1 C#Cc1ccc(CC(N2CCC(NC(C3COCC3N=[N+]=[N-])=O)C2C)=O)cc1 c1(C(=O)NCC2N(C(CC3CCC(C)CC3)=O)CC=C2)ccc2ccccc2n1 C(C(C)C)(C(O)C(=O)NCc1ocnc1C(=O)NC1CCOC12CCCC2)OC C1(NC(c2cc(OCC)n[nH]2)=O)CC2CC(NC(=O)C(C)=C(C)CC)CC2C1 C1(C)(N(C(=O)NC(CC(=O)OC)c2ccccc2)C)CC(OC)(OC)C1 C1(CNC(=NCCOC)NCc2cnc(Br)s2)CCC2(CCCCCCC2)O1 c1(C(C)C)ccc(CNC2CCN(C(=O)CC(=O)N(C)C)C2C)cc1 c1(C(N(CC(C)CNC(=O)CCC(C)(F)F)C)=O)c(F)ccc2occc12 CCC(O)(CC)CCNC(=O)CCCN(C(=O)CCCn1ccnn1)C c1(C(=O)NC2CN(C(C=CCCC)=O)CC2n2ccnn2)c(Cl)c(C)nn1C c1(OC)ccc(-c2noc(C=CCC(=O)OC(C)CN(C)C)n2)cn1 N1(C(C(=O)Nc2scc(C)n2)=O)CCC(NC(c2ccc(CF)cc2)=O)C1C C(C(C)CC(=O)NCC1CC2CC2N1C(=O)CCc1ccccc1C)OC C(=O)(C(F)C(F)(F)F)N1CCC(c2cn(CCN(C)CCS(C)(=O)=O)nn2)CC1 c1(C(=O)NC)cn(CC(=O)NCC(C)(O)CNC(=O)CCCn2cccn2)nn1 N1(C(c2nc(C)c(C)s2)=O)C2CC1CN(Cc1cnc[nH]1)C2 C=C=CCC(=O)N(CCC(=O)NC(c1nncs1)C)C(C)C C1(CNC(C(CC)(C)F)=O)CN(C)CCN1C(=O)CSc1ccc(C(C)=O)cn1 c1(C(=O)NC(C(C)NC(C(CCC)O)=O)C)ccc(CC)c(S(C)(=O)=O)c1 c1(OC)ccc(CNC(=O)C(c2ccc(C)nn2)N2CCCC2C)cc1 c1(C(N(C(c2ccc(OC)cc2)CC)CCO)=O)ccncc1N=[N+]=[N-] C1(CC(=O)N(CCCCN(C(=O)Cn2cnc(Br)n2)C)C)CC(O)C1(C)C C1(C(N2CC(CCNC(C3CC(n4cnnc4)C3)=O)C2)=O)CC1C1CCCCC1 CCCC(CC)CC(=O)NC1(CNC(C23CCC(CO)(CC2)CC3)=O)CC1 C1(C(N(CCC(C)NC(=O)CC2CC2)CC2CC2)=O)COCCN1CC(F)F C1(NC(c2n(CC)cnn2)=O)CC(C)N(C(c2cccnc2F)=O)C1 c1(C(N(CCCN(C(=O)CCOCC2CC2)C)C)=O)cc(Cl)c(Cl)n1C CC1CCCN(C(=O)C#CC(C)(C)C)C1CCNC(c1cc(F)c[nH]1)=O c1(CC(N2CCC(C(C)NC(C3CC(O)CN3C)=O)C2)=O)ccc2[nH]ccc2c1 n1(CC(=O)NCC(CNC(C(c2cnn(C)c2)OC)=O)F)nnc(=O)[nH]1 CC1C(NC(c2cnn(C)c2N)=O)CCCN1C(=O)Cc1ccn(C)c1 C(=O)(C(O)CCC(C)C)NCc1occ(C(N(C2CC(SC)C2)C)=O)n1 c1(C(=O)NC2C(NC(=O)C=Cc3cccs3)CCC2)ccc(O)c(Br)c1 C1(NC(COCCN(C)C)=O)CCCN1C(=O)CC(c1ccccc1)N(C)C.CO CCC(C)C(C#N)c1nc(C(=O)NC2CC(NC(=O)C=C3CCOCC3)C2)cs1 C1(NC(c2ncc[nH]c2=O)=O)CN(C(=O)CCc2ccnc(Cl)c2)CCC1O C1(CC=C)(NC(c2ocnc2C)=O)CCCN(C(=O)C(C)SC(C)C)C1 C1(NC(CC2CCCN(C)C2)=O)CC(F)CN(C(=O)CCCN(C)C)C1 c1(OC)ccc(C(=O)N(C2CCN(C(C3CCOC3(C)C)=O)C2)C)cc1OC c1(NC(CC)C(=O)NC2CN(CCn3cccn3)CC2(C)C)ccc(C)cc1Cl C(CC(C(=O)N(C)CC1CCCS1)NC(=O)C(F)CC1CCOC1)SC N1(C(=O)NCC2(CC)CC2)C(C(=O)Nc2cccc(Br)c2)CCC2CCCC12 c1(N2CCC(CC)C2C)nc(=NCc2cc(Br)cn2C)[nH]c2ccsc12 C(=O)(CCC(C)(F)F)NCC1N(C(CCCN(C)C)=O)CC1(C)C Cc1ncnc(C)c1C(N1CCC(NC(C2(C(=O)C3CC3)CC2)=O)C1)=O CC1CCCC(CC(=O)NC(C)CCCCNC(=O)CCc2cnn(C)n2)O1 N1(C(CCS(C)(=O)=O)=O)CC2CCCC(NC(=O)C=C3CCCCC3)C2C1 c1(NC(C2CC(CNC(C3CN(C(C)C)C3)=O)OC2)=O)cccc2cnn(C)c12.CN N1(C(c2nc(OC)oc2)=O)CCOCC12CCN(C(=O)C(C)(C)C#N)C2 N1(C(C2C(CC)CCC2)=O)CCOCCC1C(N1CCCC(C(C)(C)C)C1)=O N1(C(CCN(C(CC)CC)C)=O)CCC(CC(C)NC(=O)C(C#N)C2CC2)CC1 N1(Cc2cn(CC(=O)OC)nc2)Cc2ccccc2CC1CSc1cccnc1 CCCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(C#N)CCCCC2)=O)C1 C1(NC(CC2C(C)CCO2)=O)C2CC1CN(C(c1ccccc1F)=O)C2 C(C(C)(C)C(=O)NCC1CCC1NC(c1ccn(-c2ccncc2)n1)=O)SC C1(NC(CCC=C)=O)CC(NC(=O)CN(C)C(C)=O)C12CCOCC2 N1(C(C2(SC)CC2)=O)CCC(c2ccccc2)(NC(=O)C=C2CCN(C)CC2)C1 C1(CC)CCCC2CC12.C1(CCNC(C(C)OC)=O)(N(C(C2CC2)=O)C)CCCC1 C1(CNC(=O)C=Cc2ccoc2)CC2(CCN(C(=O)CCF)C2)CO1 N1(C(CN(C)C)=O)CC(NC(c2ccnc(-c3cc[nH]n3)c2)=O)CC2(CC2)C1 c1(CC(=O)N(c2cnn(C(=O)OC(C)(C)C)c2)CC)ncc(C)s1 C1(NC(CCOCCNC(C2CCC(C)O2)=O)=O)CC2CC1OC(=O)N2 c1(C(N2CCOCC2CNC(C2(CO)CCCO2)=O)=O)cnc2ccccc2c1 C1(C(C)(C)CNC2C(C(=O)OC(C)(C)C)OCC2)CC(=O)C12CCC2 N1(C(Cc2ccc(C)o2)=O)CCN(C(c2cnn(CCO)c2)=O)CC1C1CCC1 C1(NC(c2[nH]cc(C(=O)OC)c2)=O)CN(C(=O)C#CC(C)(C)O)CC(F)(F)C1 N1(C(CSCCOC)=O)CC(=O)CC1C(=O)NCCC1(CC(C)C)CC1 c1(COC)ccc(C(=O)NCC2(CN(C)C)CN(C(C3CCC3)=O)C2)c(F)c1F Cc1conc1CC(=O)NCC(C)(C)NC(C1CCCN1CC(F)(F)F)=O C12CC3CCCC3N1C(=O)CC1(CC1)CN2.N1(CC)CCCC1CC(N)=O c1(C(=O)NCC(C2CC2)NC(CCOCC(C)C)=O)cnc(S)nc1 C1(NC(=O)NCCC(COC)OC)CC12CCCCCC2 C1(C(=O)OC)(C(N2CCC(CCNC(=O)C3=C(Cl)CCC3)C2)=O)CC2(CCC2)C1 c1(C(N2CCN(C(CCC(=C)C)=O)CC2C)=O)oc2ccccc2c1COC C(C(O)C(=O)NC(c1nocc1C(=O)NC1CCCC1CN(C)C)C)=CC C1(O)(CNC(c2cccnc2S)=O)CCN(C(C2CCC(C(F)(F)F)O2)=O)CC1 c1(CC(=O)NC2C(NC(COCC(=O)NC)=O)CC2)cnc2c(=O)[nH]ccn12 C1(C(N2CCC(C(C)(C)NC(c3cccnc3)=O)C2)=O)CCC(C2CC2)CC1 c1(C(N2CCC(NC(C=Cc3ccc(SC)s3)=O)(CO)C2)=O)cc(Cl)ccc1F C=C(Br)CC(C)(C)C(=O)N1CCC(C)C(NC(=O)C(C)(C)SC)C1 N1(C(Cn2ncc(C)c2)=O)CCN(C(C2(C)CC2Br)=O)CC1C c1(C(=O)OC(C(=O)OC)C2CC2)coc2cc(F)cc(F)c12 c1(CC)ccccc1C(N1CCC2CC12C(=O)NCCC1COCCO1)=O CC(CC(N)=O)N=c1cc[nH]c(=NCCOC2CCCCC2)[nH]1 N1(C(c2ccc(CCCC)cc2)=O)CC(CNC(=O)C(C)C#N)C2(CC2)C1 c1(OC)cccc(OCC(=O)N(C)CCN(C(=O)C(=Cc2cccnc2)C)C)c1 C(CNC(=O)C(C1CCCOC1)OC)(C(C)C)NC(C1(CCCC)CCC1)=O c1(CC(=O)NC(CCN(C(c2ncn(CC)c2)=O)C)C)ccccc1C c1(CC)cccc(CC)c1NC(COC(F)(F)F)=O.C12C(C)CCN1C(=O)NC2 NS(=O)(=O)c1coc(C(N2CC3CC(C2)C3NC(c2cccc(Cl)c2F)=O)=O)c1 Cn1cnnc1C1CCC1C(=O)NCC1CCC1NC(C1(N(C)C)CCC1)=O N1(CC)CCC2CCN(C(N3CC4C(CCC=O)C4C3)=O)CC12.C1(=O)CN1.OC N1(C(C(C)Cc2cnc[nH]2)=O)CC2CN(C(c3ccccc3Cl)=O)CC2C1 n1(CC(N2C(C(C)NC(=O)C3=CCC3)CCC2)=O)cc(Br)c(O)nc1=O N1(C(C2=C(C)OCC2)=O)CC(C)CN(C(c2ccn3c2CCCC3)=O)CC1C c1(CCNC(N(CC(O)C(F)(F)F)C(COC)C)=O)c(C)[nH]c2ccccc12 C1(CN(C)C)CCCN(C(=O)CC2(N(C(=O)CCc3cncn3C)C)CC2)C1 C(=O)(C(C)(C=C)CCOC)N1CC(CCNC(CCCOCC)=O)(OC)C1 N#Cc1ccc(=NCC(=O)N2CCC3(CC2)CC(NC(c2cscn2)=O)C3)[nH]c1 C(CN=c1ccc2nnnn2[nH]1)C1(O)CCN(C(CC2C(C)CCCC2)=O)CC1 N1(C(CCC=C(C)C)=O)CCCCC1CN(C)C(C1(C)CCCC1)=O c1(CC(N2CCC(C(=O)NC(CCC)C3CCC3)(CC)C2)=O)cccc(O)c1F N1(CCNC(C2CCCN(C(C)=O)C2)=O)C(=O)NC(C)(C)C1=O c1(OC)ccc(CCC(N2CC(CCNCC3CCCCO3)C(C)C2)=O)cc1F CC(C)(C(O)C(F)F)NC(=O)CC1CC(O)CN1C(=O)CSCC(F)F CCC(CC(=O)N1CCN(C(c2cncc(O)c2)=O)C(C2CCC2)C1)CC(C)C c1(C(=O)NC(C(C)NC(CC(CC(C)C)C)=O)CO)cnc(O)c2ccccc12 C1(C(=O)NCCC2CC(NC(c3cnc(SC)s3)=O)C2)(CC)CC1(F)F c1(C(=O)NCC(CNC(c2cccnn2)=O)OC)cc(Cl)ccc1F C=CCCCCC(=O)N1CCC=CC1C(=O)NC(C[N+](=O)[O-])CCO C(=O)(C(C)CCNCC(C1CC1)NC(c1cccc(OC2CCC2)c1)=O)OC C(=O)(C(CNC(C)=O)CC)N(CCN(C(C(C=C)O)=O)C)C c1(NC(C(c2ccc(F)cc2)C)=O)n[nH]c2c1CCC(F)(F)C2 C1(C(=O)NC2CCN(C(C)=O)C2)CN(C(c2ccc(C(F)F)o2)=O)CC1(F)F C(=O)(CC1=CCOCC1)NC(CCC)C(=O)NC(C)C(C)(C)O C1(NC(=O)CCC2CC2(Cl)Cl)CC(O)(C2CCN(C(c3cscc3F)=O)CC2)C1 c1(NS(c2cccc(OCC(C)C)c2)(=O)=O)cc2c(cc1Br)OCCO2 N1(C(CNS(NC)(=O)=O)=O)CCN(C(=O)C=Cc2ccc(C)o2)C2CCC12 n1(CC)ncc(C(N2CCC(CC(C)NC(C3CC3C(F)F)=O)CC2)=O)c1Cl C(C(=O)NCC(F)F)(C(C)O)NC(CC(=O)NC)=O CCCC(C)(CC)C(=O)N1CCCC(CNC(C2CC(C(F)(F)F)C2)=O)C1 C=CCCC(C1CC1)NC(=O)C(C1(O)CN(C(=O)Cc2noc(CC)n2)C1)F c1(C(=O)NCC2C(NC(CC3(COC)CC3)=O)C2)cnc2cc(C)[nH]c2c1 C1(CC)CN(C(=O)C=C(C)CNC(C2(CO)CCCO2)=O)C(CC)CO1 N1(C(C(C)OCCC(C)C)=O)CC2C(CN(C(=O)CN3C(=O)CNC3=O)C)C2C1 c1(SCC(c2cnc(Cl)[nH]2)=O)cc2nc(Cl)ccc2s1 C(=O)(C(O)CCC(F)(F)F)N1CCOCC(NC(C2(CO)CCOC2)=O)C1 N1(C(=O)OC(C)(C)C)CCC2CC(C1)CN(C(=O)C(c1cccc(Br)c1)NC)C2 C1(CNC(c2cnc(OCC)s2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)C(C)C1 Cc1ccc(C(=O)NCCC(C)(C)NC(=O)CCc2cc[nH]n2)cc1S(N)(=O)=O CC1CN(C(=O)CCOc2cncnc2)CC1CNC(c1cnn(CCF)c1)=O C12(CNC(C(C(C)C)SC)=O)CC(NC(=O)C(N3CCC(O)CC3)C)(C1)C(C)O2 c1(CC(=O)NC2CC(CNC(CC=C=C)=O)C2(C)C)ccc(OC)c(F)c1 C1(F)(CNC(CC2(COC)CC2)=O)CCN(C(=O)CC2CCC(C)(C)C2)C1 c1(C(CC)NS(CCOCC)(=O)=O)ccccc1OC c1(C(=O)NC2CC(OC)CN(C(c3cccn3C)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 c1(OC)ccc(C(C)(C)CNC(N2CC(N3CCC3)C2)=O)cc1Br C1(NC(c2c(CC)cc[nH]2)=O)CCOCC1C(=O)N(C1(C2CC2)CC1)C C1(C(N(C2CCC(NC(=O)C(C#N)C3CC3)CC2)C)=O)CC2(CCOCC2)C1 Cc1cccc(SCC(N2CCCCC2CNC(=O)C(C)CF)=O)c1 C(CCN=c1cc(C)nc(Cl)[nH]1)OCCNC(C1C(OCC)C1)=O C1(NC(C2CCN2C(c2cnccn2)=O)=O)CCCCCC1O C12(C(N3CC4C(CNC(C(c5n(C)cnc5)O)=O)C4C3)=O)CCC(F)(CC1)CC2 N1(C(=O)CC2(O)CCOCC2)CCC2C(CCN2C(c2cccnc2)=O)C1 C1(CCNC(C(C)=CC)=O)CCN(C(=O)C(C)CN2CCCC2)CC1(F)F C1(NC(C2(C)CC(F)(F)C2)=O)CCN(C(c2cccc(N)c2N)=O)CC1F CN1C(=O)CSC1CC(N1CCSCC1CNC(=O)CNC(=O)NC1CC1)=O Cc1ccccc1C1(CNC(=O)CN2CCSCC2)CC1.N12CC3C(C3C1)C2=O c1(OC)c(CN2CC3CN(c4ccnc(OC)n4)CC3C2)cc(Cl)cc1Cl c1(C(=O)OC)ccc(CC)c(OCCn2c(Sc3ccccc3)nnn2)c1 N1(Cc2ccc(OC)nn2)CC2CCN(C)CC2C1.c12nnnn1C2C1CC1 c1(C(C)(C)C(=O)N2CC(CNC(c3cc(C(F)F)no3)=O)C2)ccc(F)cc1F N1(C(COCCCC)=O)CCC(N(C(=O)Cc2cc(C)on2)C)C(C)C1 C(C1OCc2ccccc21)NC(C(=O)NC(c1ccc(O)cc1)CCOC)=O C1(C(N(C2CCN(C(C3CCCN3N=O)=O)C2)CC)=O)CC(C)OC1C c1(C(N2CCC(O)(C(CNC(C(CC=C)(F)F)=O)C)C2)=O)cc(C)cc(C)c1O c1(CCC(=O)NC2CCN(Cc3cc(CC)nn3C)C2)ccc(C)nc1C CC1CCN(C(c2ccc(O)cc2)=O)CC1CC(N1CCCC1C(O)CO)=O C(CCN=c1[nH]ccn2c(C)cc(C)c12)CCSC C1(NC(=O)Cc2csc(-c3ccccc3)n2)CCCCN(Cc2ccc(Cl)[nH]2)C1 CC1(C)C(C(=O)NC2CCC(CNC(C3CCCS3)=O)CC2)CCS1(=O)=O CC(C)C(C)C(CNC(c1ccc(C#N)o1)=O)NC(c1ccncc1F)=O C1(COC)(CNC(c2cncc(F)c2)=O)CCN(C(c2cc(C)nn2C)=O)C1 c1(C(=O)NCCN(C(CC2ON=C(CC)C2)=O)CC(C)O)nc(Cl)cc(N)c1Cl N1(C(c2cccc(F)n2)C(=O)NCCCCCC)CCCC(C)CC1 C(=O)(CC1C(=O)Nc2ccccc21)NCC1(N(c2nc(CO)nc(=N)[nH]2)C)CC1 S(=O)(=O)(c1ccc2nc(N(C)Cc3ccccc3C)sc2c1)NCC=C=C C1(N)CC2(CCN(C(=O)C(C)(C)O)CC2)C1.C1(CC(C)CN)CCCCC1 Cc1nc(Cl)c(NC(C2CC3CC3N2Cc2ccc(-n3ccnc3)cc2)=O)nc1C N1(C(C(CC)F)=O)CCC(NC(=O)CN2CCCS2(=O)=O)C(CC)C1 C(=O)(C1=NOCC1)N(CC(CC)NC(C1(C(C)(F)F)CCC1)=O)C N1(C(CCOc2c(CC)cccc2)=O)CC2(CCC2CNC(C2(O)CC2)=O)C1 c1(C(c2nnnn2CC2CCCO2)NCc2nc(C)sc2)cccc(C(C)(F)F)c1 C(=O)(C1=C(c2ccccc2)SCCO1)N1CCC(NC(CC(C)OC)=O)CC1 N1(C(C2C(C)C2C)=O)CCOC2(C1)CN(C(C1CC3(CCCC3)CO1)=O)C2 C=C(C)C1CCC(C)=CC1CC(N1CC(CNC(c2ccc(NC)nc2)=O)C1)=O c1(NCCC(CCC)C)nc(N(CC(C)OC)C)nc2c1ncn2CC C(=O)(C(F)(F)CC(=O)N1CCCC1CNC(=O)COc1cc(F)cc(F)c1)NCC CC(C)CCCC(=O)NC1CC2C1CCN2C(=O)C(=O)C(C)(C)C C12(C(N3CCC(CCC)C3)=O)CC1CN(C(=O)Cc1csc(C)n1)C2 c1(C(=O)OC)ccc(C(C)Nc2ccc(OC(F)(F)F)cc2)cc1 C(CCCCC(=O)N(CC(C)NC(c1c(Br)ccnc1C)=O)C)SC N1(C(=O)Cc2nccs2)CCCC(N(C(=O)CCCOc2cccnc2)CCO)C1 C(CC)(C(=O)N(C)CC1CCN(C(C2CC3(CC3)C2)=O)C1)OCC C1(C)(CC)CCCN(C(=O)CC(C2CC2)NC(=O)C(C)n2cccc2)C1 N1(C(C(C)SCC)=O)CCCCC1C(=O)N(C)CCC1CCCC1 CC(O)C(C)(C)C(=O)NCC1(O)CN(C(c2cccc(C(N)=O)c2F)=O)C1 S(=O)(=O)(C1C(C(F)(F)F)C1c1ccc(Br)cc1)NC(COCC)C N(C(=NCCCN(C)C(C)C)NCC1CC2CCC1N(C)C2)C1CC(C)C1 C1(CN(CCOC)Cc2ccccc2)CCCN1c1nc(C)ns1 C1(CNC(C(COC)(C)C)=O)CCCCCN1C(c1cccc(F)c1F)=O c1(C(N(C(C)C)C)=O)cc(CNC(=O)C=Cc2cc[nH]c2)[nH]n1 CCC(CC(C)C)C(=O)NCC12CC(C1)C(NC(c1cnoc1C)=O)CO2 N1(C(CN2C(C)CCC2)=O)CC(C2(NC(c3cccc(C(=O)N(C)C)n3)=O)CC2)C1 N12CCCC(C1C)NC2=O.c1(OC)cc(COC(F)F)ccc1OC c1(C(N(C2CCCN(C(c3nc(C)oc3OC)=O)C2)CC)=O)cc([N+](=O)[O-])n[nH]1 N1(C(COCCN(C)C)=O)CCN(C)CC1CNC(C1CC(O)CC(=O)N1)=O C=C(C)CCCC(=O)N(C1CCCN(C(C2CC=CCO2)=O)C1)CCF CC(C)CC(C(=O)NC1COCC1O)N(C)C(c1cccc[n+]1[O-])=O C(C(=O)NC1(C(=O)NCc2ccc(C)cn2)CC(F)C1)(C(C)(C)C)OC C1(CC(=O)NC2(CF)CN(C(c3cnns3)=O)C2)CCCCC1(F)F C1(F)(C(N(CCC(C(C)C)NC(c2ccc(=O)n(C)c2)=O)C)=O)CCCCCC1 S(=O)(=O)(c1ccc2nn[nH]c2c1)NC(CC)Cc1ccc(C)cc1 c1(C(=O)NCCN(C(=O)CC2CCC(C(N)=O)O2)CC)cc(C)oc1C(F)(F)F C(=O)(CC(C(F)F)NC(=O)C(C1CCCCC1)=O)N(C)Cc1onc(CC)n1 Cc1nc(O)ccc1C(=O)NC(CC1CCOCC1)C(=O)NCC=CC1CC1 C(=O)(C(C)(C)OC)NCCN(CCC)C(c1csc(-c2ccoc2)n1)=O C1(C(=O)NCCN(C(C)C)C(C)C)CCCCCCN1C(=O)C(C)n1cccn1 C1(C)(OCC(=O)N(CC(C)CNC(=O)C=CCO)C)CCOCC1 C1(NC(C2=NOC(CONC(c3n(C)ccn3)=O)C2)=O)CCC2(CCC2)C1 CC1CN(C(=O)C=C2CCC(C)(C)CC2)CCC1N(C(=O)CN(C)C)C C(C(C(C)C(C)C)NC(=O)COc1ccsn1)NC(Cc1nc(C)[nH]n1)=O Cc1cc(C)c(C(N2CC(NC(=O)CCSCC(N)=O)C(O)C2)=O)cn1 C(=O)(C(C)C(F)(F)F)NCC(CNC(=O)CCC(=O)N1CCC(C)C1)OC CCCCCCCCC(F)C(=O)NCC(C1CCN(C(=O)CCC2CC2)CC1)(C)O Cc1conc1C(=O)NC(C)CC1CN(C(=O)C(c2ccnn2C)O)C1 C1(C(=O)NCC(C)(C)O)CCN(C(C23CC(F)(C2)C3)=O)CC1 C1(C)(C(=O)NCCCC(C)NC(c2c(C)c[nH]c2)=O)CCC(F)(F)C1 c1(C(=O)NCC(C)(C)CNC(C2CCC(F)C2)=O)cccc2nc(S)oc12 CC1=NOC(C)(C(=O)NCC2CCN(C(=O)Cc3cncc(Br)c3)C2)C1 CN1CCC(C(=O)OCC2OCCCC2(C)C)S1(=O)=O c1(CC(C(CC)CC(=O)N2CCC(NCC)C2C)=O)ccc(C(F)(F)F)cc1Cl c1(NC(C(C2CC(S(C)(=O)=O)C2)F)=O)nccc(=NCc2ocnc2C(N)=O)[nH]1 c1(NC(C23CCC(C2)C3)=O)ccc(O)cc1.C12COCC1CNC(=O)C2 Cn1ncc(C#N)c1C(=O)NCC1CC2CC2N1C(=O)CCc1cncnc1 C(=O)(C(C#N)C(C)(C)C)N1CC(N(C(C(CC)=CC)=O)C)C(O)C1 c1(C(=O)NC2CN(C(=O)C=CC3CCC3)C2)cccc(=S)n1O N1(C(CCn2c(C(C)C)ncc2)=O)CCC(O)(C(C)NC(C2(CCF)CC2)=O)C1 N1(C(C(C2CCC2)OCC)=O)CCC(O)(CCNC(=O)CSC)C1 C1(N(C(=O)C(CC2CCOCC2)NC(C2C3CC4C(C3)C24)=O)C)CCCC1C#N c1(C(N2CC(CNC(c3ccnc(Cl)c3Cl)=O)OCC2)=O)cccc(F)c1F N1(C(CCc2ccc(=N)[nH]c2)=O)CCCC2CN(C(c3cccs3)=O)CC12 N1(C(C(c2cc(C)n(C)n2)=O)=O)CCC2(CC1)CC2(F)Cl CC1CCC(C)N1CC(=O)NC1CCC(CNC(=O)CCc2nc(O)n[nH]2)C1 CC#CCC(C(=O)NC1(C(F)(F)F)CC1)NC(c1cc(COC)on1)=O c1(C(=O)NCc2n[nH]c(C)c2C)cc2sc(N(CC(C)C)CC)nc2s1 c1(-c2ccc(NC(c3cc(C)[nH]c3C)=O)c(F)c2)csc2ccccc12 C=CCCC(C)(c1nnnn1CCC)NCc1cncn1CC N1(C(c2coc(C)n2)C(=O)NCCCC)CCNC(=O)C12CCC2 N1(CC)CCN(C(=O)C(CC(C)(C)OC)NC(=O)OC(C)(C)C)C(C)C1 c1(C(=O)NC2CCCC(NC(C(C)C)=O)C2)cc2cc(N)ccc2s1 N1(CC(=O)NC2(C)CC(NC(c3c(C)onc3C3CC3)=O)C2)CCS(=O)(=O)CC1 C(=O)(CCCCO)NC(C1CN(C(=O)C=CCN2CCOCC2)C1)C C#CCS(=O)(=O)CCn1nnnc1NC1CS(=O)(=O)C1 Cc1cccc2c1OCC2C(=O)N(C(C)CN(C)C(c1cnc(O)n1C)=O)C c1(CNC2C(C(=O)NCc3ccc(Cl)cn3)CCC2)nc(Cl)ccc1Cl NC(=NCC1CC1)NC1CC1C.C12(CC)CC(C(=O)N(C)C)(C1)C2 c1(C(N(CCCNC(c2ncnn2C)=O)CC)=O)n[nH]c2c1COCC2 C(=O)(CCCN1CCCC1)NC(CCNC(CN(CCCCNC(C)=O)C)=O)C c1(C(N2CCC(N(C(Cc3nnc(C)o3)=O)C)C2)=O)cccc(NS(C)(=O)=O)c1 N1(C(c2c(N)non2)=O)CC2COCC(C1)C2NC(=O)Cc1cnns1 N1(C(C(CC)OC)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(C(C)C)C1 C(c1cccnc1)=CCONC(COC1(C)CN(C(C(C)CO)=O)C1)=O CC1(C)CC(C(=O)NCC(C)(C2CC2)NC(C2CCCC3C2C3(F)F)=O)=NO1 c1(C(=O)NC(C2N(C(c3cn(CC)nn3)=O)CCC2)C)cccc2[nH]ncc12 c1(C(=O)NC(C(C)(C)C)CNC(=O)C(F)(F)C2CC2)nccc2occc12 CCC(CC(=O)NCCC1(NC(=O)C(C)Cc2ccncc2)CC1)SC c1(C(N(C2CCCN(C(CC(C=C)CC)=O)C2)CCF)=O)ccc(F)c(C)c1Cl c1(C(=O)NCC2(C)CCN(C(C3CCCN3C3CC3)=O)C2)cccn2nnnc12 Cc1ccc(C(=O)NC2(C)CCN(C(C3CC34CC(O)C4)=O)C2)nc1 Cc1cc(F)cc(C(=O)NC(C2CN(C(C3CCC(C)CC3)=O)C2)C)c1N c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC1CN(C(=O)CC2CC(OC)C2(C)C)C1 c1(C(N(C)CCC2CCCCN2C(=O)Cc2nc[nH]n2)=O)cc2cccn2cn1 CCCCC(C(=O)N1CC(S(N)(=O)=O)C1)NC(c1cnn(C(C)C)c1)=O c1(NC(C(=O)N(CC(C)NC)C)=O)cccc(N2CCOCC2)c1C CC1(C)CC1(C#N)C(N1CCC(CNC(=O)CCNC(C2CCC2)=O)C1)=O N1(C(=O)C2=CCCN(Cc3cc[nH]n3)C2)CCc2[nH]c3ccccc3c2C1 C(C(C)(C(=O)NC1CN(Cc2cnc(-c3ccccc3)o2)C1)N(C)C)NC(C)=O C1(C(N2C(C)(C)C(NC(=O)C=Cc3ccsc3)CC2)=O)CCOC2(CCOCC2)C1 C1(C)(OC)CCCN(C(=O)C(C)(C)C2CCCN2C(=O)COCCC(C)C)CC1 n1(CC)nnc2c1C(C(=O)NCC1CC(=O)N(C)C1)CN(C(=O)CC#N)C2 C(N=c1[nH]c(=NC2CCNC(=O)CC2)[nH]c2ccccc12)C1CCN(C(C)C)C1 C=CCC(CC)C(=O)NC1CC(C(=O)NCCN2CCC(C)(C)C2)CC1O CCC(C)C(=O)NCC(=O)NCc1cn(C2CCN(C(=O)CCSC)C2)nn1 c1(NC(c2ncccc2NC(c2csnn2)=O)=O)cc2cc(F)ccc2cn1 N1(C(c2ccc(C=CC(=O)OC)cc2)C(=O)NC)Cc2ccc(O)cc2C1 N1(C(C=C(C)C(C)C)=O)CC2CC3CC2C1C3NC(=O)Cc1nnc(O)s1 c1(N(C2CCCCCCC2)C(=O)NCC2CC(C(C)C)OCC2)cnc(S)n1C C(=O)(C1=CC(C)(C)C1)NC(CC(=O)NCCc1ccc(C)nc1)C C(=O)(C(CCS(C)=O)N(C)C)NCC(N(C(C=C(C)Cl)=O)C)C1CC1 C#CC1CCN(C(=O)CCC2CCN(C(C3(CO)CCC3)=O)CC2)C1 N1(C(CCC(C)CN(C)C)=O)CCC2(C)CN(C(c3n[nH]cc3F)=O)CC12 CC1CCN(CC(=O)NC(C)CCN(C)C(c2cc(CN(C)C)nn2C)=O)CC1 C(CCCCC(=O)N1CC(C(C)NC(C2(F)CCOC2)=O)C1)OC c1(C(=O)NC2(CC=C)CN(C(=O)C(F)n3cccn3)C2)cc(F)c(CO)c(F)c1 C1(CCC)CCC(c2nnnn2C(C)C)(NC(c2cccc(F)c2)CF)CC1 C1(CNC(c2coc(Cl)c2)=O)CC12CCN(C(c1c(Cl)nsc1Cl)=O)CC2 C(=O)(C1Cc2ccccc21)N(C)CC1CCN(c2ccnc(C3CCC3)n2)CC1 c1(C(=O)OC)ccc(Br)c(C)c1C.N12CCN(CC1)C(=O)c1ncccc1C2 c1(C(N2CC(C)OC3(CCC3)C2)C(=O)NCCSCC)cc2ccccc2nc1C N1(C(c2[nH]cc(CC)n2)=O)CCN(C(=O)C(O)CN(C)C)CC12CCC2 N1(C(C2(NC(c3cc(Cl)no3)=O)CSC2)=O)CCC(C2CCOC2)C1 C1(C(=O)NCCNC(C2(C)CC2)=O)CCCN(C(C2(C(F)F)CC2)=O)C1 C1(CN(C(C(C)OCC(C)C)=O)C)COCCN1C(=O)CC1CSC1 C1(NC(C2(COC)CC=CC2)=O)CC2(C1)CN(C(c1cc(C(N)=O)cn1C)=O)C2 N1(C(COCCCCCC)=O)CCC(COC)(NC(=O)C(c2cccnc2)O)C1 C1(N(C(CCCSC)=O)C)CCCN(C(C2(P(C)(C)=O)CC2)=O)CC1 C12(CC)CCC(C(=O)NOC3CCCC3)(CC1)CO2 C(CC(O)CNC(=O)CCc1nc(C)no1)NC(C=C(C)Cl)=O N1(C(C(CC)N(C)C)=O)CCN(C(c2cc(Br)c(F)cc2C)=O)CC(O)C1 N1(Cc2nc(C)sc2)CC2(CCC(NC(c3cc(C(C)C)nn3C)=O)CC2)C1 c1(CC)nnsc1C(=O)NC1COCC1C(=O)NCCC1(C)CCCO1 c1(C(=O)NC(CNC(=O)C(=Cc2c[nH]cn2)F)CO)cnc2ncc(Cl)cn12 CCCCC(O)C(=O)NCC(C1CCCCCC1)NC(=O)CN1CC(CC)C1 Cc1ccc(C(=O)NCC(CC2CC2)C(=O)N2CC(N3CC(F)C3)C2)c(C)c1 C1(F)(C(=O)NCC(CC)NC(=O)C(C)(C)N2CCOCC2)CCC(C)CC1 CC1CN(C(c2ccc(N(C)C)cn2)=O)CC1NC(C1CCCC1CF)=O c1(CC(N2CCCC(N(C(=O)CC3(C)CC3(F)F)C)C2)=O)csc2ccccc12 C(C1CCN(C(=O)C(C)C2CC2)CC1)=CC(N1C(CN=[N+]=[N-])CCC1)=O N1(C(COCCCCCC)=O)CC2CCOCC2(NC(c2ccc(=N)[nH]n2)=O)C1 c1(CC(=O)NC(C(=O)NC(C=C)CO)C)cn(C)cn1 c1(NC(C(N2CCC(NC(N)=O)C2)C)=O)ccc(S(=O)(=O)N2CC(O)C2)cc1Br S(=O)(=O)(c1ccc(I)cc1)NC1CC(C)CN(c2ncnc3cccnc23)C1 CC1CCCCN1S(=O)(=O)Cc1csc(OC(C)(C)C)n1.N12CCN(CC1)C2=O C1(C(C)CC(=O)O)CCN(C(c2nscc2Br)=O)CC1 c1(N2CC(C)(C)C(NC(=O)C=Cc3ccccc3)C2)ncnc2cccc(F)c12 n1(NC(CC=C)C(=O)O)cc2ccc(-c3c(OC)cccc3OC)cc2n1 N12CCN(CC1)CCN(C)C(=O)C2=O.CC1CCOC1C(=O)OC(C)(C)C C(=O)(C(F)(F)C(O)C(C)C)NC(C1OCCN(C(CC(C)OC)=O)C1)C C(=O)(C(C)S(=O)(=O)C(C)C)NCCN(C(c1cc(N)no1)=O)CC N1(C(C(C)SC(C)C)=O)CCC2C(C1)CN2C(c1ccsc1Cl)=O C(=O)(C(C)CC(N)=O)NCC(c1c(OC)cccc1)NC(=O)Cc1cncnc1 N1(C(c2ccc(C#C)o2)=O)CC2CC(NC(=O)C(O)CCSC)CC2C1 Cc1cc(F)ccc1C(=O)NC1CCCC(CNC(C2CCS2(=O)=O)=O)C1 CC(CCCCNC(=O)CNC(=O)CC1CCCC1)NC(C1CCC(=O)O1)=O C=C(CNC(=O)COCCNC(=O)C(F)C1CCOC1)CC C(=O)(C(C)CC(=O)c1ccccc1F)N(CCCNC(c1cnn(C)n1)=O)CC Cc1cc(OC(F)F)c2ccccc2n1.N12CCN(CC1)CC2=O N1(C(CCC(CC)OC)=O)CC2=C(C1)CN(C(c1cc(SC)c(C)o1)=O)C2 N1(c2c(CC(=O)OCC)cnc(Cl)n2)CCC2CCN(C(=O)CO)CC2C1 N1(C(C(C)=CC)=O)CCOC(CCNC(=O)CC2(O)CCCOC2)C1 c1(C(=O)NCC(CCNC(C2CC(Cl)(Cl)C2)=O)OC)cn2c(C)cccc2n1 N1(C(c2nccc(CC)c2)=O)CCCC(NC(C2CC(C(C)C)=NO2)=O)CC1 c1(OC(C)(C)C(=O)NC2CC2NC(=O)CC2(C)CCC2)cc(Cl)cc(Cl)c1 c1(CC)nc(C)c(CNC2(c3ncc(C)o3)CC2)o1 C=C(C)C1OCCCC1C(=O)NC(C)(CNC(=O)C(=C1CCCCC1)F)C(C)C C1(N(C(C(C2CCCN(C(c3ccn(CC)n3)=O)C2)C)=O)C)CNC(=O)C12CC2 C1(CNC(=O)C=CC2CCC2)COCCN(C(=O)CC2CCOC2)C1 C1(C(=O)NCC(CNC(c2nc(OC)c(C)s2)=O)C)C2CC(F)(F)CC12 c1(C(=O)NCC(CC)NC(=O)C(C)n2cncn2)c(Cl)cccc1[N+](=O)[O-] C(C(O)C(=O)NCC(C)N(C)CC)NC(CSCCC)=O C1(C(=O)NCCC(=O)NCC(C)(O)C2(C)CC2)(OC)CCSC1 c1(C(N(CCN(C(c2c(N)cccc2Cl)=O)CC)CC)=O)nccc(Cl)c1F c1(N2CCOCC(C(C)C)C2)nc(=NC(C)CN2CCCC2)[nH]c2c1CSC2 CN1CCC(CC(N2CCC(O)C2C(=O)NC(C2CCCCC2)CO)=O)CC1 C1(NC(c2c(OCCOC)n[nH]c2)=O)CCN(C(c2cccc(OC)n2)=O)CC1 N1(C(C2CCC(CCNC(C3CC3C(F)F)=O)CC2)=O)CCN(CC#C)CC1 C1(CC)CCn2cncc2C1.C12CN(CCN1C(C)=O)C(=O)c1sc2nc1C c1(OC)cccc(CCC(=O)N(CCCN(C)C(C2(C#N)CCOC2)=O)C)c1F C1(NC(C2(SC)CC2)=O)CC(F)CN(C(=O)Cc2csc(-c3cccs3)n2)C1 c1(C(=O)NCC2CCCN2C(=O)C=CC2CCCO2)cc(F)cc2ccoc12 N1(C(c2onc(CC)n2)=O)CCC(NC(C2(C)CC=CCC2)=O)C(C)(C)C1 CC1(C)CCCC(CC(N2CCN(C(=O)CC3CCC(=O)NC3)C(CO)C2)=O)C1 CS(=O)(=O)C1CCCC1C(N1CC2CC(Nc3cc(Cl)ncn3)C2C1)=O c1(C(N2CC(c3ccc(C)s3)C2)=O)cccc(C(=O)C(F)(F)F)c1 c1(C(N2CCC3(CC2)CN(C(=O)CC2CCCO2)C3)=O)cc2cc(Cl)cnc2o1 CC1(C(N2CC(NC(C3CCC(N=[N+]=[N-])C3)=O)CC(O)C2)=O)CCNC(=O)C1 C1(NC(CCN(C)CC)=O)CC2CCC1CN(C(=O)Cc1ccc(C)s1)C2 c1(C(C(=O)N(CC(C)CNC(C2CCCO2)=O)C)(F)F)ccc(Cl)cn1 Cc1ccccc1C=CC(=O)NC1CC(C)CN(C(=O)C(C)(C)C(N)=O)C1 Cc1ccc(O)c(C(=O)NCC2CC2CNC(=O)CN2C(=O)CCCC2=O)n1 N1(C(C(C)CC2CCC2)=O)CCN(C(C2CCCC2(C)C)=O)CC(C)(C)C1 CC1(C)CC1(C(N1CC(NC(=O)C2CC2)C1)=O)CNC(C1CC=CCO1)=O C1(NC(C2CCCC23CC3)=O)CC2CCC1N2C(=O)Cc1ccccc1 O=C(NNC(=O)C(O)c1ccncc1)C1CC2(CC2)CN1 C1(N(C(C(F)=CCC)=O)C)CCCCN(C(=O)Cn2cc(C(F)F)cn2)C1 Cc1ccc(C(=O)NC2CC3CC(NC(c4c(CO)cnn4C)=O)C3C2)cc1O NC(=O)CC(O)CC(=O)N(CCNC(=O)C(F)(F)C1CC1)Cc1ccccc1 c1(OC)ccc2ccnc(C(C)NC3CC4CC3C3CCCC43)c2c1 C1(C(C)NC(c2ccc(F)cc2)=O)CN(C(=O)CCCc2nncn2C)CCO1 c1(C(=O)NCC2(F)CCC(CNC(C(C)C#N)=O)CC2)cc2ccncc2[nH]1 Cc1ncc2n1CCC(C(=O)NCc1cnc(NC(c3cccs3)(C)C)s1)C2 C1(CCC(=O)N(C(C)CN(C(=O)C)C)C)CCCOC1.c1(CC)cc(O)n[nH]1 n1(CC(=O)NC2CCCN(C(c3cccn(O)c3=O)=O)CC2)nc(Cl)ccc1=O C(=O)(C(F)CC(C)(C)C)N(CC(C)C)CC(N1CC(F)(F)C1)=O CC1(C#CC(=O)NCCC2CCN(C(=O)CC(c3ccccc3)N(C)C)C2)CC1 c1(OC)ccc(C(N2C(NC(=O)NCc3ccccc3)CCCC2C)=O)nc1Br C(=O)(C(F)=C1CCCC1)N(CCNC(CSCCC)=O)CCC c1(NCc2cccs2)nnc(-c2cnccn2)n1CC(C1(C)CCC1)OC(=N)O N1(C(C2CN(C)C(=O)N2)=O)CC2(C1)C(NC(=O)CC1CCOC1)CCS2(=O)=O N1(C(c2c(C#N)ccs2)=O)CCC2CN(C(c3ccc4ncnn4c3)=O)CCC12 C(=O)(C1(C)CCc2cc(C)ccc21)NC1CCCC(C(=O)OC(C)(C)C)CC1 C1(CNC(=O)Cc2cscn2)CN(C(C2CS(=O)(=O)C2)=O)CCO1 Cc1cc(CC(C)C(=O)NC2(c3cn(CCN(C)C)nn3)CCC2)cc(C)c1Br C1(C(=O)NC(C)CCNC(=O)CCc2ccc(O)cc2)CS(=O)(=O)CC12CC2 c1(C(=O)NC(C(C(C)C)NC(=O)CCc2cnn[nH]2)C)cnnc2ccccc12 CCC(C)(CNC(=O)CCN(CCC(C)(C)C)C)NC(C1CC(C(C)(C)C)C1)=O C(=O)(C1=COc2ccccc2O1)NC1CN(C(C(C)SCC)=O)C2(C1)CCC2 C1(CC(N2CCC(C)(CCNC(C(CCSC)O)=O)C2)=O)CCC(C)(C)CC1 C(=O)(CC(C)C(C)(C)C)NC(CC1CN(C(c2nn(CC)nc2C)=O)C1)C Cc1cc(CN(CCC(C)NC(=O)CCC)C2CC2)nn1C(C)(C)C C(=O)(C(C)CC(C)(F)F)NC1(C)CCN(C(c2ccc(OC)nc2C)=O)C1 CCCC(CCC)=CC(=O)NCC1CN(C(C2C(C)(C)C2(C)C)=O)CC1C c1(CNc2nccc(C)n2)ccnc(NC2CN(C(C(CO)OC)=O)C2)c1 C(C(=O)NCC1COCC1NC(=O)CCN1CCCC1=O)(C(C)C)OC Cc1cc(NC(=O)C(=O)NC2CCCC2Oc2ccccc2)ccc1S(N)(=O)=O N(C(=NCCNc1ccccc1Br)NC(C)C)CC(COC)F c1(CN)ccc(NC(=O)C(=O)NCC2CCNC2=O)cc1C(F)(F)F c1(C(=O)NCCN(C(c2cc(CC)no2)=O)C(C)C)cncc(C(F)(F)F)c1 CC1CN(C(=O)C(C)Cc2cnn(C)c2)CC1CNC(=O)C(C)(C)CO C#CC1(O)CCCN(C(=O)C(CN(C)C)NC(=O)Nc2cn(C)nn2)C1 c1(C(N2CCN(C(C(c3scc(C)n3)C)=O)CC2CF)=O)cn(C)c(=O)cc1C c1(C(=O)NC(COC)C(=O)NCCOC2(C)CCCC2)ccccc1F CC1CC(C)(C)N1C(=O)OC(C)(C)C.C12CCN(CC1)C(=O)CC(=O)N2 C1(CCC(=O)N(C2CN(C(C34CC(C)(CO3)C4)=O)CC2O)C)NC(=O)NC1=O N1(C(c2c(CC)nco2)=O)CCN(C(=O)CN(C)CCO)CC1C(C)(C)C Cc1cccc(C)c1OCC(=O)NCC1CCN1C(C1CCS(=O)(=O)N1C)=O N1(C(=O)CCC2CCC2)CCCC2(CCN(C(=O)CN3C(=O)CCC3=O)C2)C1 c1(OCC(C)C)ccccc1C(N1CC(n2cc(C(C)O)nn2)C(C)C1)=O c1(C(=O)NC2CN(C(c3ccc(Br)c(Cl)c3)=O)CC2O)c(O)cc(O)cc1O C1(CC=C)(NC(=O)CC2COCCO2)CCN(C(c2cccn2C)=O)C1 C1(NC(c2c(C)occ2)=O)CCCC(NC(c2ccccc2OCC(N)=O)=O)C1 c1(CNc2ccc(N(CC)CC)cc2Cl)c(C)nn2ccccc12 CN1CCCN(CCCNS(=O)(=O)CCCCl)CC1 c1(-n2c(C)nc(C(=O)Nc3cccc(-c4nc(=O)o[nH]4)c3)n2)ccc(Cl)cc1Cl C12(NC(C=CCCC)=O)CCC(CC1)N(C(=O)C(C)CCc1ccccc1F)C2 c1(CC(=O)NCCC(C)N(C)C(c2ccnc(O)c2)=O)cc(F)cc(F)c1 Cc1ccc(F)c2oc(C(=O)NC(C)C(C)NC(=O)COc3cccnc3)cc12 c1(C(C)=O)cc(C(=O)NCC2(C(=O)NC34CC(C3)C4)CC=CC2)n[nH]1 CC(CF)CC(=O)NCC(C)(C)Cn1cc(COC2CCOCC2)nn1 CC1CN(C(=O)Cc2ccc(Br)cn2)CCN1C(c1c(Cl)cccc1Br)=O C1(NC(CC2CC(=C)C2)=O)CN(C(c2ccc(OC)c(Cl)c2)=O)CC1(C)C C1(c2cc(CNC(C(C)C3CCC3)=O)on2)CCN(C(C2CCC(C)O2)=O)CC1 N1(C(c2cccc(SC)c2)=O)CCC2(CCC(NC(=O)CC3(O)CCC3)C2)C1 N1(C(C(C)=C(C)C)=O)CC(NC(C2COC(=O)C2)=O)C2(CC2)C1 C1(NC(c2ccc(Br)c(O)n2)=O)CC2CC(C1)CN(C(C13CCCC1C3)=O)C2 c1(C(N(C2CN(C(=O)C=CC3CC3)C2)C)=O)c(O)cccc1Cl CC1CCN(C(c2nn[nH]c2Cl)=O)CCN1C(=O)Cc1cccc2nsnc12 c1(NC(CCN(CCC)C(=O)Oc2c[nH]c(C)cc2=O)=O)ccc(F)cc1Cl CC1CCC(NC(C2CCC(C(F)(F)F)CC2)=O)CN1C(c1ccc(CO)s1)=O CCC(C)(C)C(C)CC(=O)N1CCC(C)(NC(=O)CCc2c(C)noc2C)CC1 c1(C(=O)NCC(CC)C(=O)N2CCCC2CN(C)C)cc(C)cc(O)c1 C1(CC)(NC(=O)CC(C)CF)CCCN(C(C2(COCC)CC=CC2)=O)C1 Cc1c(F)ccc(C(N2CC=CC(NC(=O)CCC3CCCCC3)C2)=O)c1Cl c1(C(=O)NCC2(F)CC(NC(c3n(CC)ncn3)=O)C2)cccc(N)n1 Cc1c(Cl)cnn1CC(=O)NCC1CN(C(C2CC2c2cccnc2)=O)CC1O c1(C(CN(C2CCCC2)C(C2CCN(Cc3cnccn3)C2)=O)O)ccccc1 C1(O)(C(N(CC(CN(C(CC2CC(=C)C2)=O)C)O)C)=O)CCCCCC1 Cc1ccncc1C=CC(=O)NCC1(F)CCCN(c2nccc(CO)n2)C1 C1(CC)(NC(C2(COC)CC2(F)F)=O)CN(C(=O)COC2(C)CCC2)C1 C(=O)(C1=CC2CCCCC12)N1CC2N(C(C(C)(C)CF)=O)CC(C2)C1 N1(CC(=O)N(C(C(CC)CC)C(=O)OC)C)CC(=O)N(C)CC12COC2 C=CCC(CC=C)C(=O)NCCC1CCN(C(=O)CC2(CSC)CC2)C1 C1(CNC(COC)=O)COC(C)(C)CN1C(=O)CCc1n[nH]c(=N)s1 N1(C(CCOCC#C)=O)CCC2CN(C(C3(SC)CCOCC3)=O)CC12 N1(C(C(=O)NCC)C(C2CCOCC2)OC)CCC2(CCC(O)CC2)C1 c1(C(=O)NCC2CCN2C(=O)CC2CCCC2)cc2cc(F)ccc2[nH]c1=O C1(C(N2CCC(NC(c3cc(C(N)=O)[nH]n3)=O)(CF)C2)=O)CCCC2C1C2(F)F C12(NC(c3nc(C(=O)NCC=C)sc3)=O)CCC(CC1)N(C(=O)C(C)CC)C2 c1(CC(=O)NC2C(C(=O)Nc3c(SC)cccn3)C2)cn2c(C)csc2n1 C1(C(=O)Nc2ccc(C)nc2)CN(Cc2ncn(C)n2)CCC1(F)F c1(C(N(C2CC2)CC)=O)ccc(CCC(=O)NC2CC(C(=O)OCC)C2)cc1 C1(CNC(C(C)OC)=O)CCN(C(c2cccnc2SC(C)C)=O)CC1(F)F C1(C(C(=O)OC)N(C2CCOCC2)C)CCCC2CC12.C12CC1NC2=O C(N=c1[nH]c(N2CC3CC=CCC3C2)nc2ccsc12)C1(C)CC2CC2C1 C1(C)(C(=O)NCC2N(C(c3cc(OC)ns3)=O)CCC2)C2CC3CC(C2)CC1C3 C1(C(=O)NCC(C)N(CCC(C)C)C)CCN(C(=O)C=Cc2ccoc2)CC1O CN1CCOC2CC(NC(C3CCCC(NC(=O)OC(C)(C)C)C3)=O)CC12 Cc1cc(C(=O)NCC(N2CC3(C2)CN(C(C)C)C3)=O)ccc1[N+](=O)[O-] C=CC(CCC)CC(=O)N1CCC1C(=O)NCC1CCC(O)CC1 c1(OC)ccc(C(=O)NC2CC(CNC(c3c(F)cccc3Cl)=O)C2)cc1F c1(CC)cccc(NC(c2cc(Cl)cn2C)c2nnnn2CC)c1 C1(N(C(c2c(C)cnnc2)=O)C)CCCCN(C(C2CCCO2)=O)C1 N#Cc1cccc(C2=CCCCC2)c1-c1cnn(CC(CC(F)(F)F)=O)c1 c1ccc2nc(CNC(C3=NOCC3)c3nnnn3C3CCOC3)ccc2c1 C1(C(N2CCC(O)(C(C)NC(c3c(C)coc3)=O)C2)=O)CC(C2CC2)=NO1 c1(OC)cc(OC)cc(C(=O)NC(C)C(C)NC(=O)Cc2cc(Cl)ccc2Cl)c1 c1(OCC)cccc(C(=O)NCCOCCNC(c2ccnc(C)c2N)=O)c1O C(=O)(C(C)CCN(C)C(c1ccccc1)=O)NCCNC(COCCOCC)=O C1(C)(CNC(C(c2ccccc2)N(C)C)=O)CCC(NC(=O)C(C)(C)F)CC1 N1(C(c2cncc(C#N)c2)=O)CCC2(CCCN2C(c2cnc(O)nc2O)=O)C1 C(CC1=CCOCC1)NCC1C=COC1 N1(C(CS(=O)(=O)NC)=O)CCCC2C1CCN2C(=O)C=CCOC C1(CC#C)(C(=O)NCCN(C)C(c2csnc2OC)=O)CCCC1 c1(SC)cccnc1C(N1CC2C(CNC(=O)CC(C)CN(C)C)C2C1)=O c1(OC)cc(C(=O)NCC2(C)CCCN(C(c3scnc3C)=O)C2)ccc1C C(C(C(F)(F)F)OC)NC.c1(C(OC)OC)ccc(C(C2N(CC)CCC2)O)cc1 N1(Cc2ccc(C)o2)CCC2C(CCN2C(=O)C(c2cc(Cl)ccc2Cl)(C)C)C1 CCC(C)CC(=O)NCC1(F)CCC(NC(c2ncccc2C(F)(F)F)=O)C1 C(N=c1cc(C(F)(F)F)c(Cl)n[nH]1)C1C(C(=O)OC)C1 Cc1ccc(C)c(C(N2CCN(C(C3CC4C=CCC(C3)C4)=O)CC2C)=O)c1O C1(NC(C(CC2CC2)NC(c2ccc(CC)s2)=O)=O)CC(C)(OC)C1(C)C c1(CNC(CS(CC)=O)=O)nc(CNC(=O)C(F)C(=O)OCC)cc(O)n1 N1(C(c2c(COC)nn[nH]2)=O)CC(NC(=O)C=CSC)CC12CCC2 CCCCCC(O)CC(=O)N1CCC(NC(=O)CSCC(F)(F)F)C1C CC1CN(C(=O)NCCNS(=O)(=O)CC2CCC2)CCC1Cc1ccccc1 c1(C(N2CC3C(C(=O)NCC4(COC)CCC4)C3C2)=O)cccc2ncoc12 c1(CC)cc(C(=O)NCC2CC3(CC3)CN2C(=O)C(C)N(C)C(C)=O)ccc1F c1(OC)ccc(CNC(=O)Oc2csc(OC(C(C)NC(C)C(C)C)=O)n2)cc1 N1(C(=O)OC(C)(C)C)CCN(Cn2ncc(C(C(F)(F)F)SC)c2F)C(CO)C1 c1(C(N2CCC(C(=O)NC(COC)C3(C)CC3)O2)=O)n[nH]c2ccccc12 C(=O)(C1CCCc2cncn21)NC1(CF)CN(C(C(CCC)CC(C)C)=O)C1 C(=O)(C(CCC(=O)OC(C)(C)C)N(C)C)N(CCNC(=O)CC1C=CCC1)CC c1(CSC)cc(C(N2CC(N(C)C(C34CC(C(F)F)(C3)C4)=O)C(F)C2)=O)sc1C C1(C(=O)NC2C(NC(CC=C)=O)CCC2)CCCC12CCOCC2 CCCCC(O)CC(=O)NCC(CC(C)C)NC(C1(CC(C)C)CCC1)=O c1(C(N2CC(N3CCN(C(C4(C)CC4(F)Cl)=O)CC3)C2)=O)cnc(Cl)cc1Cl CCC(C(=O)NCC1CCC1NC(C1(c2ccccc2)CC1)=O)n1nccc1C CC1(CNC(=O)CC2CC(NC(c3cncc(C4CC4)c3)=O)C2)CCCC1O C1(C(N(CC(N)=O)C)=O)CC1C1CN(C(C2(F)CCOC2)=O)C1 c1(C(=O)NC2C3CN(C(C(CC)(CC)OC)=O)CC32)cc(C)cc(F)c1N c1(OC)ccc(C(C)C(N2CCCCC2CNC(c2ccn(C)c2)=O)=O)cc1F N1(C(C2(c3ccc(-c4c(SCC)ccc(F)c4)cc3)CC2)=O)CC2CCCCC2C1 C(=O)(C1=CS(=O)(=O)CCC1)NC1C(NC(CC2CN(C)C2)=O)CC(F)(F)C1 C1(C(=O)NCCN2CCCCCC2)CN(C(=O)CCc2ccccc2)CC12CC2 c1(C(=O)NC(C)CCCNC(=O)CC2CC=CC2)cc(F)c(Cl)cc1Cl N1(C(C2C(C=C)C2)=O)CCC2(CCN(C(c3ccc(OC)nn3)=O)C2)C1 c1(C(N2CC(NC(c3cncc(NC)c3)=O)C(C)C2)=O)ccc2c(c1)nnn2C N1(C(=O)OCC)CC(C(F)(F)F)(NCC(C)(C)n2cccn2)C1 CN1C(C(N2CCn3ncc(C(=O)O)c3C2)=O)CC2CCCCC12 N1(C(c2c(COC)ccs2)=O)CCCCC12CC(NC(c1nn(C)c(C)c1Cl)=O)C2 C1(CNC(=O)Cn2cc(C3CC3)nn2)CCCN(C(=O)CC2CCC(=O)N2)CC1 N1(CCCNC(c2nnnn2CCCF)C(c2ccccc2)C)CC(=O)NC1=O c1(CC(=O)NC2CCC(Cn3cc(C(C=C)(C)O)nn3)C2)ccc2occc2c1 N1(C(CC2(C=C)CCC2)=O)CC(OC)C(NC(C2(F)CC2)=O)C1 CN1CCN(C(C2CCCC2n2cccc2)=O)CC1CNC(c1ccoc1Cl)=O C#CCCCC(=O)NCC1CCCC1NC(=O)C(C1CCOC1)OCC c1(CN(C)C(=O)NCc2ccc(Cl)cc2)cc(Cl)ccn1 C1(NC(Cn2ncc(C#N)c2)=O)CC2CCC(C1F)N2C(=O)CCCC(F)(F)F C1(N(C)C(C2(C)CC2(Cl)Cl)=O)CCN(C(=O)CCc2ncc[nH]2)CC12CC2 CC1(C(=O)NCCC2(C(=O)NC3CC3C3CC3)CC2)CCNC1=O C1(C(N2CC(C(=O)NCSCCCNC(C)=O)OCC2)=O)CCn2ncnc2C1 C1(C(=O)NCc2scc(CNC(Cc3c(CC)con3)=O)n2)CC2CCCC2C1 c1(C(N(C2CN(C(=O)C(F)(F)c3cccnc3)C2)C)=O)nocc1Cl S(=O)(=O)(c1ccc(NCc2ccc(SC(F)(F)F)s2)c(F)c1)NC1C(C2C(C)C2)C1 C(=O)(CCCS(N)(=O)=O)NC(c1nc(C2CCCCN2C(=O)CCCCC#N)n[nH]1)C c1(C(C(=O)NCc2ccc(C3(C)CC3(F)F)cc2)N)c(F)cccc1F C1(NC(C(C2CCCC2)SC)=O)COCC1CN(C(=O)CCCc1cnn[nH]1)CC c1(-c2nc(-c3c(OC)ccc(O)c3)on2)c(F)ccc2ccoc12 C(=O)(CCCCC(C)(C)C)N1CC(N(C(=O)CC2CCC(=O)O2)C)C2(C1)CC2 N1(C(C(CC=C)C)=O)CC2CCOCC2(NC(C2CN3CCN2CC3C)=O)C1 c1(C(N2CC(SC)C(NC(c3cc(C#N)c[nH]3)=O)C2)=O)cc2ccc(C)cn2c1 N1(C(C#CC(C)C)=O)CC(C)(CNC(c2cncc(C(C)(C)C)c2)=O)CC1(C)C Cc1onc(C2CC2)c1C(=O)NC1CCC(NC(=O)CN(C)CCO)C1 C1(NC(c2c(C(C)C)cccc2)=O)CCN(C(=O)COC2CC2)CC1(C)C C(=O)(CC(C)C(C)(C)NC(=O)CN=[N+]=[N-])NC(c1n(CC)ncn1)C N1(C(C(C2CC2)NC(C2CS(=O)C2)=O)=O)CCN2CCCCC1C2 Nc1cnc(Cl)c(C(N2CC(CNC(c3c(Cl)csc3Cl)=O)C2)=O)c1 c1(OCC)cccc(C(=O)NCC23CC(C2)C(NC(=O)CCF)CO3)c1N C(CC(C)C)(C(=O)NC(C)(CNC(c1cnc(C)[nH]1)=O)C1CC1)OC C1(CNC(C23CC(n4cc(C5CCC5)nn4)C2C3)=O)CCS(=O)CC1 c1(CC(=O)NCCCC2OCCN(C(c3n(C)ccc3)=O)C2)nc([N+](=O)[O-])n[nH]1 Cc1cnccc1C=CC(N1CCC(N(C(=O)CC2CCCCO2)CCO)C1)=O C1(CCNC(=O)Cn2cccn2)CN(c2ccncn2)CCS1(=O)=O CCC(C)C(C(=O)N1CC2CC2(C(=O)NC(C2CCCO2)CC)C1)NC(N)=O c1(N(C2CCC(NC(C3(C(F)F)CCCC3)=O)CC2)C)cc2nncn2cn1 CC(C)(C)S(=O)(=O)c1ccc(C(=O)Nc2cnc([N+](=O)[O-])c(Br)c2)cc1 N1(C(CCN(C(C=CC(=O)N(C)C)=O)C2CC2)=O)CCOC(C)C1CCCO c1(C(=O)NC2CC(NC(CCC)=O)C23CCC3)cc(Br)c(C)cc1O CC1(C)C(NC(c2c[nH]c(C(N)=O)c2)=O)CC1O CN(C)NC(=O)CCC(=O)NCC1CN(C(c2ccsc2C(F)F)=O)CCO1 c1(CCC)nc(C(=O)N(CC(C)N(C)C(c2coc(Br)n2)=O)C)cs1 C(CCO)(C(F)F)NC(c1c(C(C)NC(=O)C(C)C2CCCC2)noc1)=O C(c1ccc2c(c1)CCO2)=CC(=O)NCCCCCNC(C(C(=O)NC)(C)C)=O c1(SCC2CC2)cc(C)c(CCNC(c2cccc(NC(=O)OC)c2)=O)cc1Cl Cc1c(C(N2CCC(C(F)C(=O)NCC3C4CCCCC34)C2)=O)cncc1F c1(C(=O)NCC2(C)CCC(NC(C=C(C)C3CC3)=O)C2)cn2c(C)csc2n1 CC1CCC(CNC(C2CCC2NC(C2(C)CC(F)(F)C2)=O)=O)CC1 Cc1nc(CN2CCCCC2c2ccc(Br)nc2)c(F)c(Cl)n1 N1(C(c2c(Cl)ccc(OC)c2)=O)CCOC2CN(C(=O)Cc3ccsn3)CC12 CS(=O)(=NC(=O)C(F)(F)CC(=O)N1CCOCC1)c1ccccn1 Cc1cc(C(=O)OCc2ccnn2CCF)c(C)nn1 CC1CCN(C(c2ccncc2Cl)=O)CC1NC(C1(NC(N)=O)CC1)=O c1(C(=O)OC)nccc(C)n1.N1(C(C2(C(=O)OC)CC2)=O)CCC1C(C1CC1)N C1(C)(COC)CC(NC(c2oc(CO)nc2C)=O)CN1C(C1CN(C(C)=O)C1)=O C1(C(=O)NCC(CCCC)NC(c2cc(O)nc(O)c2)=O)CCC2CC2CC1 c1(C(=O)NC2C(C(=O)NCCOCCC)C2)csc(C)c1 N1(CCCCOC(C)C)CCCC2C(NC(C3CC(O)C3)=O)C(C)(C)C12 C#CCC(C(=O)N1CCCC(OC)C1)NC(c1ccncc1O)=O C=CC(CC)CC(=O)N1CC2(CC(CNC(=O)C(C(C)C)SC)C2)C1 Cc1nn(C)cc1CCC(=O)NCCN(C(c1cc(C2CCC2)on1)=O)C1CC1 C1(C)(NC(C(c2ccc(F)cc2)SC)=O)CCN(C(c2cc(F)c[nH]2)=O)C1 C(CCCC(C)NC(=O)CCC=C(C)C)NC(c1c(CC)cno1)=O C(=O)(CCc1ccc[nH]1)OCC1C(C)C1 C1(O)(C(C)OC)CCN(C(C2C(C)(C(=O)OCC)C2)=O)CC1 n1(CC(C)C)nccc1C(=O)NCC1(CNC(=O)C(C)(C)n2cccn2)CCC1 c1(C(=O)OC)cc2cc(C(=O)NC3COCC3n3cc(C4CC4OC)nn3)sc2s1 CN1CCOC2(CN(C(C3CN(C(c4nc(Cl)cs4)=O)CC34CCC4)=O)C2)C1 C1(CNC(C2(C#C)CCC2)=O)CCC12CCN(C(=O)CC(C)(O)C(F)(F)F)CC2 c1(CNC(c2scc(-c3cc(OC(C)C)ncc3)n2)=O)nc(Cl)ccc1Cl C1(CNC(=O)Cc2ccc(O)nc2)CCCN(C2CCOCC2)C1=O C(=O)(C1COc2ccc(Cl)cc21)NCC1(C)CCCN(C(C(C=C)(C)C)=O)C1 N1(C(CN2CCN(C(C)=O)CC2)=O)CC2CCC1CN(C(c1scnc1C)=O)C2 c1(OCC)ccccc1CC(=O)N1CCC1CNC(c1sc(C(C)C)nc1C)=O C1(F)(CC)CCCN(C(=O)CC(C(F)F)NC(=O)CC2CCC2)C1 CC(C)CC(C)(O)CNC(=O)C(CO)NC(=O)CCNN(C)C c1(OC)cc(CC(=O)OCC(c2cc(F)cc(Br)c2Cl)=O)cc(Br)c1OC c1(OC)c(C(=O)NC2CN(C(C3CCCCC3)=O)CC2C(F)(F)F)ccnc1Cl N1(CC(N2CCC(CNC(COC(CC)C)=O)(CO)C2)=O)Cc2ccccc2C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2(N(C)C)CC2)=O)cn(C)c(=O)nc1O C12(C(=O)NCC(C)(C3CC3)NC(C(C=C=C)C)=O)CC3CC(CC1C3)C2 c1(OCC)ccc(C(N2CC(NC(c3cnn(C)c3)=O)C(CC(C)C)C2)=O)cc1 c1(NC2C3CN(C(C4C(C)OC(C)C4)=O)CC2C3)ccc(Cl)cc1[N+](=O)[O-] C1(CNC(c2c(C)scc2)=O)CCN(C(c2ccc(F)cc2Cl)=O)C(C)C1 C12(NC(c3ccnc(CO)c3)=O)CC3CCC(C1C2)N3C(=O)Cc1ccsc1 C(CNC(c1[nH]nnc1C)=O)(CC(F)(F)F)NC(c1cc(OC)ncn1)=O C(=O)(CC1=CCCC1)OC(C1(C)CC2CC2C1)=O.N12CCC(O)C1C2=O C(C1CCCCC1)=CC(=O)NCC1CN(C(=O)C=C2CCCCC2)CC1O N1(C(=O)OC(C)(C)C)C2CN(C(=O)NC(c3ccc(Cl)cc3)C(F)(F)F)CC12 C1(COC)(NC(c2ccc(F)cn2)=O)CCN(C(C2CC(n3ccnc3)C2)=O)C1 C1(C(C)OCC)CCN(C(=O)C(C2(O)CN(C(=O)OC(C)(C)C)C2)F)CC1 C1(NC(C2C3(CC(C)(C)C3)C2)=O)CCCCC12CCN(C(C1(F)CC1)=O)C2 c1(CN(C2C(C)CN(C(=O)CC(C)C(F)F)C2)Cc2nccs2)nn(C)c2c1CCC2 c1(C(C(=O)OC(C)(C)C)N(C)CCN(C)CCC2CCOC2)coc(Br)n1 Cc1c(C(N2CCC(C)C(NC(C3(C(C)C)COC3)=O)C2)=O)[nH]c2ccccc12 c1(C(=O)NCCN(C(c2csc(-c3cn[nH]c3)n2)=O)CC2CC2)cscc1F CC(CF)CC(=O)NC(C)CC(C)NC(C1CC(OC(F)F)C1)=O CC1CCN(C(c2ncc(F)cn2)=O)CC1NC(=O)CCC1CCCCC1 CCC(C)CCCC(=O)N(CC(C)N(C)C(c1c(C)cc(C)cc1C)=O)C C1(CN(C(c2c(CC)onc2)=O)C)C2CN(C(=O)CCN3C(=O)CCC3=O)CC12 CCC(O)C(C)C(=O)NC1CCN(C(C2CN(c3nncs3)C2)=O)CC1F C(=O)(C(F)C(C)(C)O)NCC(CNC(c1c(C)nn(-c2cnn(C)c2)n1)=O)CO c1(NC2CC3CN(C(C(C)C(C)(F)F)=O)CC32)nc2c(cc1C#N)CCOC2 N1(C(c2c(C)noc2C)=O)CCN(C(=O)Cc2ccccc2)C2(CC2)C1 C1(C(N(CC(N2CC(C)=C(C)C2)=O)C)=O)CCCCC1(C)C Cc1ncnc(N2CCCC(CN(C)C(C3CCCC(C(N)=O)C3)=O)C2)c1F C1(C2(NC(C(C3CCC3)OC)=O)CC2)CCN(C(c2cnccc2OC)=O)CC1 CC(C)(C#N)CCCC(=O)N1CCC(C(=O)NC2CC3C(C2)C3(F)F)C1 C12(C(N3CC(O)(CNC(=O)C(O)C4CCCC4)C3)=O)CC(C1)S(=O)(=O)C2 C=CC1COCCN1C(C1CC(O)(CNC(=O)CC2C=CCCC2)C1)=O N1(C(CN(C(=O)CC2OCCCO2)C(C)=O)=O)CCC2CCCCC2C1 C(CCCC(C)NC(c1cccc(=O)o1)=O)NC(c1c(C)cns1)=O N#Cc1cccc(C2=NC3CCCN(Cc4cccc(F)c4F)C23)c1 N1(C(c2ccc(OC)c(Br)n2)=O)CC(N(C(=O)CC(C)OC)C)C2(CC2)C1 C=CCC(CC)C(=O)N1CCN(CC2(NC(c3ccc(CC)cc3)=O)CC2)CC1 C(=O)(C(C(=O)OC(C)(C)C)C(C)(C)C)NC1CC(C)(NC(C(C)SC(C)C)=O)C1 c1(-c2n(-c3cnc(C)s3)nc(C3CCCO3)n2)ccc2nc(Cl)nn2c1 c1(NCc2cnc(CC)[nH]2)cc(N2CCC(OCC(F)F)C2)nc(COC)n1 N#CC1CC2(CC(N3CCN(CC(c4nc5ccccc5[nH]4)=O)CC3)C2)C1 c1(C(=O)NC2(CCNC(CC3COCC(C)O3)=O)CCC2)csc2nccn12 N1(C(Cc2cn(C)nc2)=O)CCC(C)(C)C1CNC(C1CC(F)C1)=O C=CC(C)(C)CC(=O)NCCN(C(=O)C(C)(C)OC)C C12(CC)CCC(C(N3CCC(O)(CNC(=O)CC4COCC4O)CC3)=O)(CO1)C2 C(=O)(C(C)S(C)(=O)=O)NCCn1cc(C(N(C(CC)C)C)=O)nc1 C#Cc1cccc(C(C(=O)NCc2ccco2)N(C(C)CCO)C)c1 C1(F)(CNC(C(C)N2CCCC2)=O)CCN(C(c2ccc(Cl)cc2)=O)C1 N1(C(C(CCCC)NC(c2cc(Cl)n[nH]2)=O)=O)CCc2cccc(F)c21 CCN(OC)C(=O)CCN(CCCNC(=O)CCNS(=O)(=O)c1ccccc1)C C12(c3n(CC(=C)C)c(N(C)Cc4cc(C(C)C)no4)nn3)CCCCC1CCC2 C(C(CC(C)C)C(=O)OC)CCC.C#CC1(C(=O)O)CCCC1 Cc1nn(C)c(C)c1CC(=O)NCCC(C)N(C(=O)CN1OC(C)(C)CC1=O)C C1(NC(c2ccc(Br)c(F)c2)=O)COC2(CCN(C(=O)CO)CC2)C1 c1(CC)cc2c(N3CC(CC(=O)Nc4ccnc(CC)n4)C3)ncnc2s1 C1(CNC(CN(C)CC)=O)CC(NC(c2ccon2)=O)C1 c1(CNC(=O)NC(c2ccncc2Br)CC(=O)OC)nccc(Cl)c1F CC(CS(C)(=O)=O)C(=O)N1CCN(C2CN(C(C3CCC(=O)CC3C)=O)C2)CC1 c1(C(N2CCC(CN(C)C(C3(CC4CC4)CCC3)=O)C2)=O)noc2c1CCCC2 C(=O)(C1=C(Cl)CCCC1)NC(CN(C(c1c(CC)nn(C)c1)=O)C(C)C)C c1(CNC(C(=O)NCCCOC)=O)ccc(Br)cc1OC(F)F c1(C(=O)NCC23C(CN(C(C(CCC)NC(N)=O)=O)C2)C3)c(OC)ncnc1C n1(CCCC)nccc1C(=O)NCCCN(C(c1ccc(COC)s1)=O)C1CC1 c1(C(N2CCC(NC(C3(O)CC(F)(F)C3)=O)CC2)=O)ccn2c(O)nnc2c1 CC1CCC(F)(F)CN1C(C1CCC2(CC2)N1C(=O)C(Cl)Cl)=O c1(C(=O)NCCN(CCC)C(C2CCCCO2)=O)ccc(CS(N)(=O)=O)cc1 C(=O)(C(F)C(F)(F)F)NCc1cn(CC(C)NC(=O)C(C)(C)F)nn1 C1(CNC(C2(C)CCCN2)=O)CN(C(C2(O)CCOCC2)=O)CCO1 c1(CC)ccccc1C(N1CCC(O)(CNC(=O)CCc2ccsc2)C1)=O N1(C(C(C)OC2COC2)=O)CCc2ccccc2C1CCNC(C1(Br)CC1)=O C1(F)(CNC(CNS(N(C)C)(=O)=O)=O)COCCN(C(c2nonc2N)=O)C1 c1(C(C(=O)NCC(C)C)N(C(c2ccc(F)cc2)(C)C)C)cccc(C#N)c1 c1(CCCCC(=O)N(CC#C)C)ccc2c(c1)OCCO2 N1(C(=O)C2=CCCCC2)CCC(NC(C23CCCN(CC2)C3)=O)C(F)(F)CC1 N1(C(C2C=C(C)CS2)=O)CC(CC(=O)NCCOC2(C)CCC2)CC1(C)C c1(C(N(C(C)C)CCN(C)C(C23CC(C)C2C3)=O)=O)ccc2c(c1)CCNC2=O c1(C(=O)NCCC(CNC(=O)Cc2csc(S)n2)O)cnn2c1CCC2 Cc1nccc(C(=O)N(CC(O)CNC(C2(c3nc[nH]n3)CC2)=O)CCO)n1 CC1ON=C(C(=O)NCC2(C)CN(C(=O)CCP(C)(C)=O)CCO2)C1C C1(NC(c2c(CC)n[nH]c2)=O)CCC(F)(CNC(c2cncc(C(F)F)c2)=O)C1 C1(C)(OCC(=O)NCCCC(C)NC(C2(CC=C)CC=CC2)=O)CCOCC1 N1(C(C2CC(OC)C2)=O)CCC1(C)CC(=O)NCc1nc(N(C)C)n[nH]1 CC1(C)CC(CNC(c2cnns2)=O)CN1C(C1CCCC12CCC2)=O c1(-c2cn(CC(CC)O)nn2)cc(C(N2CCOC(C3CC3)C2)=O)c(F)c(F)c1 Cc1[nH]nc(C(=O)NCC2CC(NC(c3sccc3F)=O)C2(C)C)c1Cl C(CCC1CC1)(C(=O)N1CCCC1CF)NC(CCNC(=O)OC)=O CCC(CC(=O)N1CC(C(N2CCCC2CC(C)C)=O)(COC)C1)C(C)(C)C C(=O)(CCCCCOCCO)N1CC(NC(C(c2ccc(F)cc2)C)=O)C1 c1(C(N2CCC(C(C)CNC(=O)Cc3cn[nH]c3)CC2)=O)cccc2ccoc12 N1(Cc2ccc(OC)c(Cl)c2)CCC(NC(c2coc(C(F)F)n2)=O)C(C)(C)C1 c1(C(=O)NCCC2CCN(C(CNC(=O)OCC)=O)C2)cccn2cnnc12 Cc1cccc2c(C(N3CC(C4CN(C(c5cnn(C)c5)=O)C4)C3)=O)c[nH]c12 C1(CNC(c2c(C(C)C)occ2)=O)CC2(CCC2)CN1C(=O)C(C)C1CC1 C1(C(=O)NCC2(CC(=O)NCCC(=O)NC(C)C)CC2)CCOCC1(C)C C1(COC)(CNC(C2CCC(=O)NC2)=O)CCCN1C(=O)CN1C(=O)CCC1=O c1(CC(N2CC(NC(C=C(C)Cl)=O)C3(C2)CC3)=O)ccc2oc(O)nc2c1 c1(C(N(C2CCN(C(=O)CC(C)OC)CC2)CCCC)=O)cc2c([nH]1)CCOC2 N1(C(COC)=O)CCC2(CCCC2NC(=O)CC(O)CN(C)C)CC1 C1(CCNC(c2c(CCNC(C(CO)OC)=O)n[nH]c2)=O)CCC(C)(C)O1 c1(CNC(C23C(CN(C(=O)NCC(=O)OC)C2)C3)=O)ccc(Cl)c2ccccc12 CC(C)C(F)(F)CC(=O)NCCOCCCNC(=O)C(c1ccccc1Cl)C c1(C(=O)NCC(C)NC(C(CC#C)O)=O)ccc([N+](=O)[O-])c(OC)c1 C(CCC1CC1)(C(=O)N1CCCC1C(C)NC(=O)C(C)OCC1CC1)OC N1(C(C(C(COC)C)C)=O)CC2CCCC(NC(=O)Cn3nc(C)oc3=O)C2C1 CCCCC(O)C(C)C(=O)N1CCC2(CCC2)C(NC(=O)C(O)CSC)C1 C1(C(=O)NC(CCCNC(c2c(C)nc(C)s2)=O)(C)C)CCOC2(CCCC2)C1 c1(CC(=O)NC)csc(C2CCCN2C(=O)OC(C)(C)C)n1.C=C1CC1C(=O)O CN(C)S(=O)(=O)NCC(=O)NCC1CCC(NC(c2ccccc2F)=O)CC1 C(C(C)(C)C(=O)NC1(C)CC(NC(=O)C(F)F)C1)NC(=O)OC(C)(C)C C=CCC(C(=O)NC1CC12CC(NC(c1ccccc1C#N)=O)C2)C(C)C c1(OC)cccc(CC(=O)NC(CNC(=O)Cc2cccnc2)CO)c1 CC1CCC(NC(=O)CS(N)(=O)=O)CN1C(c1cc(Cl)cnn1)=O C(C(C(=O)NCC1CC(O)C1)C(C)(C)C)NC(C(C)C(F)F)=O C12(NC(=O)Cc3ccno3)CCN(C(c3cc(O)nc(O)n3)=O)CCC1C2 N1(C(c2ccc(C)nc2C)=O)CC(NC(=O)C(C)c2ccco2)C(C2CC2)C1 C1(CC(=O)NCC2CCN2C(=O)CCc2ncc[nH]2)CC2(CC2)C1 C1(NC(CCSCC)=O)(CO)CCN(C(c2cc(O)cc(F)c2)=O)CC1 CC(C(=O)N1CC(CC(=O)N(C2COC(C)(C)C2)C)(N(C2CC2)CO)C1)C(F)(F)F N1(C(c2c(C)ccc(C(N)=O)c2)=O)CCC2(CC1)CN(C(C1CCC1(F)F)=O)C2 CCCC(C(O)C(=O)NC1(C)CC2CCC1C2)NC(=O)CCc1cscn1 CS(C)(=O)=NCC(=O)N1CCCC1C1CCN(C(=O)Cn2cnc(C(N)=O)n2)C1 c1(C(N2C(C3CCN(C(C(=C)F)=O)CC3)CCCC2)=O)cc(F)c(Cl)c(F)c1 c1(NC(C2CCC(CNC(CC3(C)CCCO3)=O)C2)=O)cc(=O)n2ccsc2n1 C(=O)(CCCC(C)C)N1CC(C#C)(C(=O)NOCCOCCF)C1 C1(C(N2CC3(CC(NC(C=C(CCC)C)=O)C3)C2)=O)OCC2CCCCC12 N1(C(C=CSC)=O)CC2CN(C(c3cnc4n(c3=O)CCS4)=O)CCC2(CO)C1 c1(C(N(c2ccc(NC(C3(C4CC4)CC3)=O)cc2F)C)=O)cc(Cl)c(Cl)cc1N C1(NC(=O)CC2CC2(Cl)Cl)CCN(C(c2cc(Br)co2)=O)CCC1CO N1(C(C(N2C(C)CCC2C)C)=O)CCN(C(=O)CCC2OCCO2)CC(C)(C)C1 CC(N=c1nc(N2CCn3nc(C4CC4)cc3C2)c2c([nH]1)CCS2)C1CCC1 N1(C(Cn2c(=N)[nH]nc2)=O)CCCC(O)(CNC(=O)COc2cccnc2)CC1 c1(OCC)ccc2c(c1)CCCN2C(c1cnn(CCO)c1C)=O C1(NC(C=Cc2ccc(CC)o2)=O)CCCC(NC(=O)CCS(N)(=O)=O)CC1 C(C(CO)(CO)CO)NC1CC(C)CNC1 C1(NC(c2c(Cl)ccc(C)c2)=O)CC2CN(C(=O)C(N)=O)CC2C1 c1(OC)nc(C)ccc1C(=O)Nc1cc(-c2nn[nH]n2)ccn1 C(C(C)(COC)C(=O)NCCn1cc(C(=O)NCc2cnc(C)cn2)cn1)OC c1(CC(=O)NC(C2CCCCC2)C(=O)N(C(C=C)C)C)cc(C)on1 c1(C(=O)NCCCNC(CC2CCCC(C)(C)CC2)=O)c(Cl)cc([N+](=O)[O-])cc1Cl Cc1nn(C)c2sc(C(=O)NCC3CCN(Cc4ccc(Cl)cc4F)C3)cc12 CC1(C(=O)NCc2ccccc2CNC(C23CCC(C2)C3)=O)CCC(=O)N1 C1(CC(=O)NCCCCNC(CCc2n(C)c(S)nn2)=O)CCCC(C)(C)O1 CCC(CC(=O)N1CCC(O)(CNC(c2csc(O)n2)=O)C1)C(C)(C)C c1(C(N2CC(C)C(CCNC(C3COC4(CCC4)C3)=O)C2)=O)c(N)cccc1F C(=O)(CCC(C)N(C)C)NC1(CCNC(c2c(C)con2)=O)CCC1 c1(NC(C)=O)ccc(CC(=O)NC2CN(C(=O)CCOC3CCC3)C2)cc1Cl C=C(C)CC(C)C(=O)NCc1ccc(CNC(C2(CC)CC(F)(F)C2)=O)cc1F Cc1nc2c(C(N3CC4CCN(C(=O)CC(C)CN(C)C)C4C3)=O)ccnc2[nH]1 C(CC(C)C(=O)N1CC2CC2(CNC(=O)CC23COC(CF)(C2)C3)C1)OC N1(CC)CCN(C(=O)CC2CN(C(C3CC4(CCC4)C3)=O)CC2C)CC1 c1(C(c2n(CCCC)nnn2)NCC2COCCO2)cncc(Br)c1C CC(C)CC(C(=O)NC(C)C(C)(C)NC(c1ccc(C2CC2)cn1)=O)C(C)C CC1(C)OCC2CC12C(=O)NC1CC(NC(c2cnc3sccn23)=O)C1 c1(CC)ccc(NC(=O)CC2CCCN2C(=O)COCCCOC)cn1 c1(C(N(CC(CNC(CC2C(C)CCO2)=O)(C)C)C)=O)cc([N+](=O)[O-])cn1C CCC(CNC(=O)CCNC(c1cc(Cl)ns1)=O)C(C)(F)F c1(C(=O)NC2(CCO)CN(C(CC(C=C)C)=O)C2)cnc(O)c(C(F)(F)F)c1 n1(C(C(=O)N(C(CNC(CNC(=O)OCC=C)=O)C)C)C)nc(C)cc1C c1(C(=O)NC(CNC(C=CCC)=O)CC(C)C)cc(C)cc(Br)c1F CC1CCN(CCC(=O)NCC2(F)CC(NC(=O)C(C)NC(N)=O)C2)CC1 C(CCCCCC(=O)NCC1CC2CCC(C1)C2)NC(C(C)C1CC1)=O C1(C(NOCCCC#C)=O)CCN(C(c2cnnn2C(C)C)=O)CC1(C)C C1(NC(COC(C)C)=O)CCC2CN(C(=O)C(C)(C)C(C)O)CC2C1 N1(C(C2=CC(C)(CC)C2)=O)CC2CN(C(c3cc(C)ccc3NC)=O)CCC12 N1(C(c2c(C(=O)OC)con2)=O)C(CNC(C2(CO)CCCO2)=O)CC2CC12 c1(C(=O)NC2(CNC(C3C(C)(C(C)C)C3)=O)CCC2)nccnc1N C1(C(=O)NCc2ncc(C(=O)NC(C)Cc3cccnc3)[nH]2)CCNC(=O)C1 c1(OC)ccc(Br)cc1C(N1CCC(C)(C(=O)NCC2(C)CC2)C1)=O C(C1(O)CCc2ccccc21)NC(CC)C1CC1C Cc1nc2ccc(C(=O)NNc3noc(C4CCOCC4)n3)cc2o1 c1(C(=O)NC(CNC(C(c2ccc(CC(C)C)cc2)C)=O)C)ccc(N)cc1F C(C)(CNC(C1CCC(C(N)=O)C1)=O)(C(C)C)NC(c1cnc(CCC)s1)=O c1(C(=O)NC2CN(C3CN(C(CC4(C=C)CC4)=O)C3)C(=O)C2)cc(F)ccc1C c1(NC(CCC)=O)ccc(NC(=O)Cc2ccc(Cl)c(OCC)c2)c(C)c1 C1(NC(CCNC(C)=O)=O)CCOCC1NC(=O)CSc1nnnn1C Cc1ncoc1C(=O)NC1(CCNC(=O)C(=O)Nc2ncc[nH]2)CC1 C1(C)(CNC(C2C(CC)CCN2C(=O)CNC(=O)OCC)=O)CCC(O)CC1 C1(C(=O)C)CCN(C(=O)C(N2CCCC2C(C)(C)O)=O)CC1.CO c1(C(=O)NC2CCCN(C(=O)Cn3cnc(Br)c3)CC2)ccc2ccoc2c1 c1(C(=O)NCCOC2CCN(C(c3cc(C)[nH]n3)=O)C2)c(Cl)ccc2c[nH]nc12 c1(-c2nnc(N(CC=C)C)n2CCC(=O)NC(C)C)nc2c(s1)COCC2 CC1(NC(C2CC2[N+](=O)[O-])=O)CN(C(=O)C(F)CC2CCOC2)C1 N1(C(CC2ON=C(C)C2)=O)CCC(C)(C)C(NC(=O)CN(C2CCCC2)C)C1 C12(NC(CCCC)=O)COC(CNC(=O)C(C)SC(C)C)(C1)C2 C1(C(=O)NCC2CCN(C(=O)CC3OCCO3)CC2)CCC2(C1)CC2(F)F N1(CC(=O)NCC(C)(O)CNC(=O)C(F)C2CC2)C(=O)c2ccccc2S1(=O)=O c1(C(=O)NCC23C(CN(C(c4cc(C)no4)=O)C2)C3)coc(S(N)(=O)=O)c1 COn1cnc(C)c1C(=O)NC1CC2(C1)CN(C(C13CCC1C3)=O)C2 c1(CC)cnc(C(=O)N(CC(O)CN(C(=O)C(c2ccc(C)s2)C)C)C)nc1 N1(C(C2C(CNC(CNC(=O)OCC)=O)C2)=O)CCC2(CSC2)C1 C1(NC(C(C)OCC=C)=O)CC2CC1CN(C(C1(CF)CCC1)=O)C2 O(NC(=O)C(C)c1ccn(C)n1)C(CC)C N1(C(C(=O)OC)C(c2ccccc2)OC)CCCOCC1(C)C.n1(CC)ccnc1CC N1(C(Cn2cc(C(C)=O)nn2)=O)CCOC2CN(C(=O)Cc3ccon3)CC12 CS(=O)CCC(=O)NCC(C1CCCCC1)NC(c1cnc(C(C)(C)C)s1)=O c1(OC(C)=O)ccc(CN2CCCC(C(=O)NCC3CCOCC3)C2)cc1 C1(NC(c2c(C)cc(C)o2)=O)Cc2ccccc2N(C(C2CC(C)(F)C2)=O)C1 N1(CC)CC(C(=O)NCCC2(O)CN(C(c3ccn(C)c3)=O)C2)CCC1=O N1(C(C2CC(CCC(N)=O)C2)=O)CC(C)(CN(C)C(=O)OC(C)(C)C)C1 N1(C(C(CSC)(C)C)=O)C2CCC(C2)C1CC(=O)NC1CC(N2CCCC2)C1 Cc1ccc(C)c(OCC(=O)NC2CC23CC(NC(c2cc(CO)[nH]n2)=O)C3)c1 C1(C(=O)NCCOCCCNC(C2(CC(=O)OC)CC2)=O)CCn2cncc2C1 c1(OC)cccc(C(=O)NCC2CCN(Cc3ccc(O)cc3Cl)C2)c1OC C(=O)(CC(C)(C)CNC(=O)CCOCC)NC1CCC(CC)CC1 C=CC(CCC)CC(=O)N1CCC(N(CCOC)C(C2CC=CCC2)=O)CC1 Cc1cc(C)c(C(N2CCOC(CNC(=O)Cc3nc[nH]n3)C2)=O)cc1N Cn1cc(CC(=O)NC2(C)CN(C(C34CC3C4)=O)C2)cn1 c1(C(=O)OC)ccc(C(N2CCC(N=[N+]=[N-])C2)=O)c(C)c1 N1(C(c2cnc(CC)s2)=O)CCC12CN(C(c1cscc1C1CC1)=O)C2 c1(OC)ccc(C(=O)NCC2CC(C(=O)N(C(CF)CF)C)C2)s1 N1(C(=O)C=CCn2cncn2)CC2(C1)CN(C(c1cccc(O)c1Cl)=O)C2 c1(CC(N2CCC(N(C(c3ccn(CCCC)n3)=O)CC)C2)=O)ccc(F)c(Br)c1 C(=O)(C(C)(COC)CC)N1CCC(C(CNC(c2ccc(CC)[nH]2)=O)(C)O)CC1 Cc1c(F)ccc(-c2nc(Sc3ccc(NC=O)cc3)cs2)c1F.C(C)(C#N)O c1(CNC(C)=O)cccc(S(=O)(=O)N(C)C)c1.c1(C2C(=O)N2)ccccc1C C1(CN(C(=O)C(F)n2ccnc2)C)CCCN(C(=O)CCc2cc(Cl)no2)C1 CC1(CCC(=O)NN2CCC(C3CC3)CC2)CCCN1C(C1CCOC1(C)C)=O N1(C(c2c(C)ccc(OC)n2)=O)CC2CCC(CNC(=O)Cc3ccsn3)C2C1 C(CCC(C)C)(c1n(C(CC)C)nnn1)NC1(CCCOC(C)(C)C)CC1 N1CCc2oc(C)nc2C1.C(=O)(CCC(=O)C(c1cc(CN)[nH]n1)=O)NCC C12CCC(C1)C(=O)N1CC(C1)Cc1cn2nn1.C1(CC)CCCN1C(C)C C(=O)(C(C)C(F)(F)F)NCCC(CC)(C)NC(=O)CC1CC=CCC1 C=CC1(CC(=O)NCC2CCCC(OC)C2)CN(C(=O)Cn2ccc(C)n2)C1 C(=O)(CCCCC(F)F)N1C(C)CC(CNC(Cc2c(C)nc(C)s2)=O)C1 C1(CC)CN(C(=O)CS)CCC1NC(c1cc(Cl)c[nH]1)=O.C(C)(C)(C)OC(=O)N(C)C N1(C(Cn2c(C)c(Cl)cn2)=O)CC2(CCCC(CNC(=O)CCC(F)F)O2)C1 CC1CC(CNC(c2cc(N)c(F)cn2)=O)CCN1C(C1CC1C(F)(F)F)=O C1(NC(=O)CC2CCCC2)CC(F)CN(C(=O)Nc2cccc(Cl)c2Br)C1 N1(C(C2(C)CC2Br)=O)CCOC2(CCC(NC(c3ccc[nH]3)=O)CC2)C1 CC1CN(C(C2CCCC(O)C2)=O)CCN1C(=O)C1=CCSC1 c1(NC(C2COCCN2Cc2c(O)cccc2F)=O)ccc2nc[nH]c2c1 N1(c2nnc(-c3[nH]c(=NC)sc3)n2CC2CC2)CCC(CO)C12CCC2 CCCC(C(=O)NCc1nocc1C(=O)N(CC(=O)OC(C)C)C)OCC N1(C(c2cc(-c3ccccc3)[nH]n2)C(=O)NCCSC)CCCC(CN(C)C)C1 Cc1scc(C(N2CCCC2(C)CNC(=O)CC2CCCO2)=O)c1N CNS(=O)(=O)NCC(=O)NCC1CC1CNC(=O)C(C)(C)OC c1(OCC(=O)NC2CCCN(CC(C)C)C2)cc2c(cc1F)CCC2NC(C)=O c1(C(C)(C)NC(CCCCO)=O)ccc(F)c(Br)c1 C123CC1CN(C2)C3=O.c1(C(=O)OC)ccc(C(=O)NC2(CCOC)CC2)[nH]1.N(C)C N1(C(c2nc(CNC(C(C(C)C)SC)=O)oc2)=O)CCN(C)CC1C C(=O)(C1Cc2c(Cl)cccc21)NC1CC(F)(CNC(=O)CSCC2CCCCO2)C1 N1(C(C(=O)NCC)=O)CCCC2CCN(C(=O)CC(=O)N(C)C)CC12 c1(C(=O)NCC2N(C(C3C(CC)C3)=O)CC(O)C2)cc2n(n1)CCO2 c1(C(=O)NCC2C(NC(CCC(C)(C)N(C)C)=O)C2)cn2cccc(F)c2n1 C1(NC(CC(C)c2cccnc2)=O)CCOCC1NC(=O)CCn1cccn1 N1(C(N2CCC(Cn3ncc(C)c3)C2)=O)CC=C(c2cccc3ccccc23)C1 Cc1ccc(Cl)c(OC(C)C(=O)NCC2CN(C(=O)CC3(CO)CC3)CCO2)c1 N1(C(C(CC)C#N)=O)CC(NC(=O)Cc2cccc(Cl)c2Cl)CC1(C)C CC(C)(C(=O)NCC1(O)CC(CNC(=O)CC2CCCCC2)C1)C1CCC1 COn1cnc(C)c1C(N1CCC(C(F)(F)F)C(NC(C2CN(C)C2)=O)C1)=O CC1CCCN(C(=O)C=Cc2nccs2)C1CNC(=O)Cn1cnnc1 C1(NC(C2N(CC)CCC2)=O)CC2CC(NC(=O)CCOC(C)=O)C1C2 C(CC(=O)N1CC(OC)C2(C1)CN(C(=O)C=C(C)Cl)C2)(C1=CCCC1)OCC c1(CC(C)C)c(C(=O)NC23CC2CN(C(=O)CC=C(Cl)Cl)C3)cnn1C CC#CCC(C(=O)NCc1cc(CC)no1)NC(c1ccon1)=O C(CCC(=O)NCC1CC1CNC(c1cc(C(C)(C)C)no1)=O)=C(C)C C#CC1(O)CCN(C(C)C(=O)NCC2CCN2C(c2snc(Cl)c2Cl)=O)CC1 Cc1ncncc1C(N1CC2C(CNC(=O)C=CC3C(C)C3(Cl)Cl)C2C1)=O C(=O)(CCP(C)(C)=O)N1CCC(C(N2CCC2C(C)O)=O)(OC)C1 C1(C(N2CCN(C(c3c(F)ccc(C)c3)=O)C3C2C3)=O)Cc2cccc(C)c2O1 N1(C(c2n[nH]c(CC)c2C)=O)CCN(C(C2CC2C2CC2)=O)CC1CO C1(NC(CCCCCCC)=O)CS(=O)(=O)CC1N=c1[nH]nc(C(N)=O)s1 c1(C(=O)NCC(C)NC(C2COCCN2C)=O)ccc2c(c1)OCC2 N1(C2C3CN(S(=O)(=O)c4[nH]cnc4Br)C(C3)C2)CCCC(C2CCC2)C1 c1(C(=O)NCC2CN(C(C3CC3C(F)(F)F)=O)CC2O)cc2ccc(F)cc2o1 C1(F)(C(=O)NCCC2N(C(C(CCSC)OC)=O)CCCC2)CCCN(C)C1 C1(NC(C(CC)n2cncn2)=O)CN(C(=O)Cc2nc(C)no2)CC1OC C=CCCC(C(=O)NC1(C2CCCO2)CC1)NC(c1nnc(S)n1C)=O C1(COC(C(COCC=C)c2ccccc2)=O)CCC2COCCC2O1 N1(C(C(C)OCC=C)=O)CCC(CC)(NC(=O)C(c2c(C)nn(C)c2C)C)CC1 c1(C(C(=O)NCC(=C)C)N(CC(C)CC)CC)cnn(C(C)C)c1I N1(C(C2CCC(OC)C2)=O)CCCCC12CCN(C)C2 C1(NC(CC(n2c(C)cc(C)n2)C)=O)CC(C)CN(C(=O)CCSCC(C)C)C1 c1(NC(c2cc(-c3ccc(C(F)(F)F)nc3)cs2)=O)c(Cl)cc(Br)cc1Br Cc1cccnc1CCC(=O)N(c1nccc(C(F)F)n1)C(C1CCC(N)C1)=O Cc1cc(C)n2ncc(C(N3CC4CCC(C3)C4NC(C3CC(O)C3)=O)=O)c2n1 c1(C(N(C(C)C(=O)NC(c2ccco2)CO)CCC)=O)cc(C)nc(C)n1 c1(C2(C(N3C(CCNC(C(C)OCCCC)=O)CCC3)=O)CC2)ccccc1Cl N1(CC)CCC(N=c2[nH]c(N3CCCC(C(N)=O)C3)nc3cccnc23)CC1C CC(C)C(N=[N+]=[N-])C(=O)NC(C)(C)CCN(C)C(C1CCC(=O)N(C)C1)=O N1(C(C2N(C(c3c(C)n[nH]c3)=O)C3C(C2)C3)=O)CCCC2(CNC(=O)O2)C1 C1(CC(=O)OC)CN(C(=O)Nc2cnc(C3CCOCC3)nc2)CC1C CC(CC(=O)NC(CNC(=O)C1=CCOC1)CO)C(F)(F)F O=C(CCC(F)(F)F)NCCC1CCCN(Cc2cc3n(n2)CCC3)C1 O=C(C1CCCc2ccnn21)NC1CN(C(=O)C=CCF)CC12CCOCC2 N1(C(C=CC=CC)=O)CCC=C(C(=O)NCC2CC(O)C2(C)C)C1 N1(c2ccc(C(N)=O)nn2)CCCC2CCC(F)(F)CC12 C=CC(CC)C(=O)N1CCC(C)(CNC(=O)CC(=O)NC2CC2)C1 N1(C(c2scc(C(N)=O)c2)=O)CCCC(CNC(c2ccc(CO)cn2)=O)CC1 C(=O)(C(CN(C)C)C(C)C)NC(CC)CNC(=O)Cc1ccc(N(C)C)cc1 C(CC(CC)C(=O)NCCCC(C)(C)NC(c1nsnc1O)=O)=CC C1(C(N(C)CC2(O)CCN(C(C(=O)NCC)=O)CC2)=O)CCc2n[nH]cc2C1C C=CCCC(CC(C)C)C(=O)NCC1CCCC(CNC(c2csc(C)n2)=O)C1 C12(C(=O)NC(CNC(C3(CC)CCC3)=O)CC(C)C)CC(C1)S(=O)(=O)C2 c1(C(=O)NCCCN(C(C2C(=C)CC2)=O)C2CC2)cnc(C)nc1C c1(C(=O)NCCC(C)N(C(=O)C2=CCCO2)C)ccccc1Cn1ccnn1 C1(CNC(CC(C)(C)C(F)F)=O)CN(C(=O)CSC2CC2)CCC12CCOCC2 c1(CC(=O)NCCC2CCCN(C(=O)CCCC3CC3)C2)cnn2c1CCCC2 CC1CN(C(c2cnsc2)=O)CC1NC(=O)CCCNC(=O)C(C)(C)C c1(C(N(CCNC(c2sccc2Cl)=O)C2CC2)=O)c(Cl)cccc1Cl CCC(C)CC(C(=O)N1CCCOC(CC)C1)NC(=O)C(C)=C(C)C C(=O)(C1CCc2cc(Cl)ccc21)N1CC(O)(CCNC(c2cc(C)oc2)=O)C1 C(=O)(C(O)C(C)(C)CC)NCC(CNC(c1c(CCCC)ocn1)=O)F c1(NCCCOC(C)(C)C)nc(N2CCC(CS(C)(=O)=O)C2)nc2scnc12 c1(C(N2C(C(=O)NC3CCC3COC)CC(OC)C2)=O)ccn2cc(C)nc2c1 C1(NC(=O)CCc2ccccn2)CCC2(CC1)CC2NC(C1CC2CC1C2)=O N1(C(C2CC(CC)(CC)C2)=O)CC(NC(=O)C(C)N(C)C)C2(CCC2)C1 C1(NC(CCCC(=O)N(C)C)=O)CCN(C(C2CC3CC3C2)=O)CC(O)C1 c1(NC(C2C(C(=O)Nc3c(C)cnc(C)n3)C2)=O)nc(C)n(C)c1C#N N1(C(C(C(C)C)CC2CCCC2)=O)CC(C2CN(C(=O)CCF)C2)C1 CP(C)(=O)C1CCC=C1C(=O)N1CC2CC1CC2NC(=O)CNC1CC1 c1(C(N2C(C(N3CC(F)(C(=O)OC)C3)=O)C=CC2)=O)cc(Br)ccn1 N1(S(C(C)C)(=O)=O)CCC2(CCN(C(=O)Nc3ccc(F)c(F)c3)C2)C1 Cn1cc(S(=O)(=O)NCC(=O)NC(CNC(=O)C(F)C2CCC2)CO)cn1 C(CCC(C)C)(C(=O)N1CCC1)NC(c1cncc(NC)c1)=O CC(C)(C)CC(F)C(=O)N1CCC(C)(CNC(c2cc(O)c(O)c(O)c2)=O)C1 C(=O)(CCCCc1cn(CCCC(=O)O)nn1)NC(CCC)C C1(OC)CN(C(c2c[nH]nc2Cl)=O)CC1NC(=O)CSCC1CCCO1 N1(C(c2c(C)c[nH]c2CC(N)=O)=O)CCCC2(C1)OCCO2 N1(C(c2cc(NS(C)(=O)=O)ncc2)=O)CCC(NC(C2CCCCS2)=O)C(O)C1 C(=O)(C(C(C)(C)C)NC(C1CC(F)C(=O)N1)=O)NCC(CCC)OCC C(=O)(CC(C)(C)C(F)(F)F)Nc1occ(C(N)=O)n1 c1(C(C(=O)NCCN(C(C2CCC(C)O2)=O)C)C)ccc(Cl)c(Cl)c1 c1(OCCOCCCOC(N2CC3(CO)CCC2CC3)=O)ccc2c(c1)CCC2 O=C(C#CC1CCCCO1)NCCC1(O)CN(C(=O)C2=COCCC2)C1 c1(CNCC2N(CC)CCC2)cc(=NC(C)CCCO)[nH]c(C(C)C)n1 CCC(CC(=O)NCCN(C(=O)C(CC1CC1)OC)C1CCCC1)C(C)C c1(CC(=O)NC2C3CCN(C(CCN(C)CC)=O)C32)ccc2c(c1)OCO2 n1(CCOC)nnnc1C(C(C)CC1CCCCC1)NCCF N1(CC(=O)NCc2onc(C)n2)CCC(F)(F)C(CNC(c2ccc(C)s2)=O)C1 c1(C(=O)OC)cc(NC2C3CN(C(=O)CCC(C)CC)CC23)cc2c1CCC2 Cc1cc(C)c(C(=O)N(CCCCN(C(=O)C(C(C)C)NC(N)=O)C)C)c(O)n1 N1(C(CC=C(C)C)=O)CCCCCC(NC(=O)C(C)(C)c2ccsc2)C1 Cc1cc(C(=O)NCCCCNC(=O)COc2c(F)cccc2F)cc(C)c1C C1(C2(O)CCC2)(C(=O)NC2C(CNC(c3cc(C(C)C)no3)=O)CCCC2)CC1 CC(CCNC(=O)CCc1ccc[nH]1)N(C(=O)CNS(N)(=O)=O)C c1(NCC(C(C)C)(C)NC(C2CC=CCC2)=O)cc(C(F)(F)F)nc2ncnn12 C(C(CC)(CC)C(=O)NC1CN(CC(F)F)C1)NC(COCC(=C)C)=O CC1CN(C(=O)C(C)(C)C(N)=O)CCC1N(C)C(c1cc(Cl)ccn1)=O c1(C(N2CC3C(NC(=O)C4=CCCSC4)C3C2)=O)ccc2cnccc2n1 C1(c2n(C(CC)C)nnn2)(NC2CC(NC(=O)OCC)C2)CC2(CCNC2=O)C1 C1(CCCNC(=O)OC(C)(C)C)CCN(CCCCCn2ccnc2)CC1 Cc1cc(=NCCC2C(C)CCCN2C(=O)CN2CCC(C)(O)C2)c(C#N)c[nH]1 C(CCF)(C(=O)N1CCCCCO1)NC(c1cnn(C)n1)=O c1(N(C2(C(=O)OCC3CC(C)C3)CCC2)C)cccc(Cl)c1Br N1(C(C(C)OCC(C)C)=O)CCC(CF)(NC(=O)CCc2cnc[nH]2)C1 C1(CCNC(CCOCCOC)=O)(NC(C2CCCC(F)C2)=O)CCOCC1 C1(C(=O)Nc2ncc(C3C(C)OCC3)s2)CCC2(CCCC2)C1 N1(C(C)=O)CC(O)CC1C(=O)NCCC1CCCN(C(=O)COCP(C)(C)=O)C1 C=C(C)C(C)(C)C(=O)NC1CCCC1NC(C1CC12CC(F)(F)C2)=O N1(C(C2(OC)CCC2)=O)CCC(C)(CC(N2CCCC2CNC(C)=O)=O)C1 C1(F)(C(=O)NCC(C2CCCC2)NC(CSCC(=O)OC)=O)CC=CCC1 C(=O)(C(CCN(C)C)NC(=O)CC1CC1)NC(CC(=O)OCC)C C1(N(C(c2ncc(C)cc2F)=O)C)CC2CCC(C1)N2C(C1(CO)CCCC1)=O c1(CC)cnn2ccc(C(=O)N(C(C)CCNC(=O)C(C(C)C)SC)C)nc12 C=CC1OCCC1NC(c1c(F)cnn1CC)c1nnnn1CCCC C1(c2n(CC=C)nnn2)(NCCc2ccc(Cl)s2)CCOCC1 C1(NC(c2c(C)nc(C)[nH]2)=O)CCC2CN(C(=O)CC3CC3C)CC2C1 CC1C(=O)N1CCN(C)C.C(CCO)SCCCN.C(C)(C)(C)NCCN C12(C(=O)NC(C(=O)Nc3ccc(OC)nc3)(C)CSC)C(=O)C3CC1C2C3 c1(C(=O)NC(C)CNC(C2CCCN2C(N)=O)=O)c(Br)nc2n1CCOC2 Cc1[nH]c(C(N2CCCC(O)C2)=O)c(C)c1C(=O)Nc1ccc(C2CC2)nc1 C12(C(N3C(C(=O)OC)CC3C)=O)CCN(C(=O)C=CC(F)F)CCC1C2 N1(C(c2c(C)cns2)=O)CCC(C(=O)NCCCC2(C)CC2)CC1 C(=O)(C(C(C)C)NC(C1(F)CN(C(C2CC(N(C)C)C2)=O)C1)=O)OC c1(C(N(CC(C(=O)N(CC(F)F)CC#C)C)C)=O)cc2cccnc2[nH]1 c1(C(C(N2CCC(N)C2)=O)=O)ccc(Cl)c(N(C)C)c1.C(C)(CC1CCC1)SC C1(C(=O)OCCn2c(C)ccn2)CC(=O)N(c2ccccc2F)C1 Cc1cc(NC(=O)NC(C)CNS(C)(=O)=O)cs1 C1(NC(C(CCOC)NC(c2c(N)cccn2)=O)=O)CCC(C2CC2)C1 C(=O)(C1=CC2CC=CCC12)NCCN(C(=O)Cc1cc(Cl)cc2c1OCC2)C c1(CNC(c2c(NCc3c(C)csc3)c[nH]n2)=O)n[nH]c2ccc(Br)cc12 c1(COCCCNC(c2nc(OCC)sn2)=O)cccc(C)c1.C1C(=O)O1 Cc1nnc2n1CC(C(=O)NCC1CCCCC1NC(C1CCCO1)=O)CC2 c1(OC)ccc(C)c(C(N2CCN(CCCNC(C3C(C)C3C)=O)CC2)=O)n1 c1(CN2CCN(S(CC(=O)NCC)(=O)=O)C3C2C3)cc(OC)c(O)c([N+](=O)[O-])c1 CC(C)C#CC(=O)NN(SN1CCOC1=O)CCn1ccnc1C(C)C C1(NC(c2c(NC)cccc2)=O)CCN(C(c2ccc(OC)cc2C)=O)CC1C Cc1cccn2ncc(C(N3CC(CNC(C4CCCC(=O)O4)=O)C(O)C3)=O)c12 c1(CNC(C(CCc2cnn(C)c2)NCC(=O)OCC)=O)ccc([N+](=O)[O-])cc1 C1(CC(=O)NCC(C)N(C(=O)Cc2ccon2)C)CCCS1 c1(CC(=O)NC(C)CCN(C)C(C2(CO)CCC2)=O)ccc2n[nH]cc2c1 C(CC(O)C(=O)N1CCC(CO)(CNC(=O)OC(C)(C)C)C1)N(C)C Cc1cc(C(N2CC(CNC(=O)CC3CCOCC3)C(O)C2)=O)cc2nc[nH]c12 Cc1ccc(O)c(CN2C(C(=O)O)CCC2C(C)(C)C)c1 C(CCCN=C(NCC1CC2(CCOCC2)O1)NC1CCS(=O)(=O)C1)OC(C)C C#CC1CN(C(c2cccnc2)=O)CCN1C(C1CC1F)=O S(=O)(=O)(c1ccc(Br)c(C#N)c1)NC(C(=O)NCc1c(SC)cc(C)cc1)=O CCC(CC)CC(=O)N1CCOCC1CN(C(=O)C(c1ccc(F)cc1)C)C CC1C(N=c2nc(N(C)CC3CCN(C)CC3)c3c([nH]2)CCCC3)CCS1(=O)=O C#CC1CN(C(c2cc(CC3CC3)on2)=O)CCN1C(c1ncnn1CC)=O C(=O)(C1=CCCCC1)NC1C(CN(C(CC(=O)OCC)=O)C)CCC1 N1(C(CC2N(C)CCC2)=O)CC(C(=O)NCC2CCCS2)CCC1(C)C N1(C(C=CC=CC)=O)CC2OCC(NC(=O)Cc3ccnc(Br)c3)C2C1 CC1(C)CC(C)(C(=O)NC(C2CCN(C(c3ccccc3C3CC3)=O)C2)(C)C)C1 C1(C)(CC(=O)N(C2CN(C(c3cnc(C(C)(C)C)[nH]3)=O)C2)C)CC1(F)F C(=O)(C1COc2ccccc21)NCC1(F)CCCN(C(COCC(=C)C)=O)C1 C12(CC(=O)NCC3CCC(CNC(=O)C=CCc4cccs4)C3)CCC(CC1)C2 C1(CNC(CCC#CC)=O)CN(C(c2cscc2C)=O)CCC1C c1(NC2(CCC)CC2)ncc(C)cc1S(=O)(=O)N(C)Cc1ocnc1C(F)(F)F c1(NC(CC2CC(C(=O)NC3(C)CCOCC3)C2)=O)cc(I)cc2[nH]ccc12 c1(C(=O)NC(CN(C(c2cc(C)c(Cl)s2)=O)C)C)ccc2c(c1)CN(C)C2 N1(C(=O)CN2CCCC2=O)CCC(F)(C(N2CCCCC2C2CCC2)=O)CC1 C1(CNC(C=CC(=O)OCC)=O)(NC(=O)CC2COCCO2)CCOC1 N1(C(C(CC)O)=O)CC2CCCC2(CNC(=O)C2=CCCCC2)C1 C(=O)(CC=CCNC(=O)CCNC(C1CCCC1)=O)OCC c1(NC(C(CNC(C2CCN(C)C2)=O)(C)C)=O)ccc(C#N)cc1O C1(NC(=O)OC(C)(C)C)CC(O)CN(Cc2ccn(C3CC3)n2)C1 N1(C(C23CCN(C(c4cccc(C)c4)=O)C2C3)=O)CCc2cc(F)cc(C)c21 C(C)(CC(=O)NNc1ccccc1[N+](=O)[O-])n1cc(CNC)nn1 N1(C(C(C)O)=O)CCCCC(Nc2cc(C(F)F)ncn2)C1 c1(C(N(C2CCN(C(C(C)CC(C)(C)C)=O)CC2)C)=O)cc2cc(F)ccc2o1 c1(C(CN(CCC)C)O)sc2ccccc2c1Cl C1(C(=O)NCC2(C)CCN(C(C3(F)CCCCC3)=O)C2)SC2C=CC1CC2 N#Cc1cccc(C#CCOC(C2CC(O)CN2C(c2ccccc2)=O)=O)c1 C(CCCCN(C)C(C1CCCS1)=O)NC(C1C(C)C1C)=O N1(C(=O)CC2COCCO2)CC2CCN(Cc3nc(Cl)ccc3Cl)CC2C1 CC(C(F)C(=O)N1CCC(NC(C2CC3CCCC(C2)C3)=O)C1C)C(F)(F)F C1(CCNC(CCSCC)=O)CCCN(C(c2cn(C)nc2C(F)(F)F)=O)CC1 C(=O)(NN1C(=O)NC(C)(c2cccs2)C1=O)c1[nH]cc(C(=O)OC)c1 c1(NC2(C#N)CCN(Cc3nccc(N(CC)CC)c3)C2)ccc2ncccc2c1 C12(NC(C=CC)=O)CCCC1N(C(c1cc(F)c(Cl)cc1OC)=O)CC2 C1(CNC(c2cnccc2Cl)=O)CC2CCC(C1)N2C(=O)CC1CCC1 C1(CN(C)C(N)=O)CCN(C(=O)NCCC2COCCO2)C1 C1(C2(NC(c3cn(C4CC4)nn3)=O)CC2)CCCN1C(C1CC1CF)=O c1(CNC(C2CC(OC)C2)=O)ccc(CNC(C2(C(C)C)CCC2)=O)cc1 S(=O)(=O)(c1cc(C(=O)NC2CCCC(C(=O)NC3(CO)CC3)C2)co1)NC C1(OC)C2CCN(C(=O)COC(C3CCCC3(C)OC(C)=O)=O)CC12 c1(OC)ccc(C)c(C(=O)NC23CC2CN(C(=O)COCc2nc(C)no2)C3)c1 C1(C2CCCC2)(C(=O)OC)CCN(S(=O)(=O)c2cnn(-c3ccccc3)c2)C1 CC1CCN(C(=O)Nc2cn(-c3ccnc(Cl)c3F)nn2)C(C)C1 c1(OC)cccc(F)c1CC(N1CC2CC1CN2C(c1ccc(O)cc1F)=O)=O Cc1c(C(=O)NCC2CC(O)CN2C(C2CC(N(C)C)C2)=O)[nH]ccc1=O N1(C(CCSCC)=O)CCC(O)(CN(C(=O)C(C)(C)N(C)C)C)CC1 c1(-c2n(-c3c(C)cccc3C)nc(C(C)O)n2)ccnc2c1cnn2C C1(NC(CSCC)=O)CN(C(c2ccc(C3CCC3(C)C)cc2)=O)CC1(C)C C(=O)(CCCCCC)NCCC(CNC(=O)CCc1cnc(C)s1)OC c1(C(N(CCN(C(=O)C=CC(=O)NC)CC)CC)=O)conc1C1CC1.N(C)(C)C CCCCCC(C)CC(=O)N(C1CCN(C(=O)C(CC)(CC)CO)CC1)CCO CC1=C(C(=O)NC(CO)C(C)NC(=O)C(C)(C)C)CCO1 c1(OC=O)ccc(OC)cc1.c1(OC)cscc1C(N1CCC(O)C1)=O.C1CN1.C1CC1 N1(C(C)=O)CCC(C)(C)CC1N(CC1=NOC2(CCC2)C1)C(=O)C(N)=O c1(NC(=O)Nc2cccc(NC(C3C(C)COC3=O)=O)c2)nc2ccccc2s1 C1(NC(C2CC3(CC3)C2)=O)CN(C(C2CC23CCCC3)=O)CC12CCCC2 c1(C(=O)NCC2C(C)(C)C(NC(c3n[nH]cc3F)=O)C2)ccc2c(c1)COCC2 C1(NC(C(C)=CC2CC2)=O)CCCC12CN(C(C1COC(=O)N1)=O)C2 C1(CC(C)O)CCN(C(C2CCCC2CNC(C23CCC(C2)C3)=O)=O)CC1 CC1(C)C2CN(C(C34CC(NC(C5C6CCC7C(C6)CC57)=O)(C3)C4)=O)CC12 N1(C(C(C(C)O)C)=O)CC2(CCN(C(C3CC(=O)C3)=O)C2)C1 N1(C(C=CCCC)=O)CCC2(CO)CN(C(C3CC4(C3)CC(C)C4)=O)CC2C1 C(=O)(CCCC(=O)N1CCCC1CC(N1CC2C=CC2C1)=O)OC(C)(C)C c1(C(=O)NC2CCC(CCNC(C(F)OC)=O)C2)cccc(CC#N)c1 C1(C)(CCC)C(=O)NCCN1C(c1cc(Cl)ccc1CNC(=O)OC(C)(C)C)=O N1(C(C(CCCCC)O)=O)CCC(NC(c2ccnn2C(C)C)=O)C2(CCC2)C1 C1(=CCCN(C(c2ncc(C(F)(F)F)[nH]2)C(=O)NCC2CC2)C)CCC(C)(C)CC1 Cc1ccc(C(=O)NC2CCCC2CNC(c2cocn2)=O)c(Br)c1F N1(C(=O)C2=CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)CC(O)(C2CCC2)C1 N1(CC)CCC(CNC(C2(CO)CCN(C(=O)Cc3cnc[nH]3)C2)=O)CC1 C(C(CO)(CO)NC(=O)CC(C)SC)N(C(c1nc(OCC)oc1)=O)C C1(CC(=O)NCCCCCNC(C2(C)CCC2)=O)C2CC3CC(C2)CC1C3 C(=O)(CCCCNC(=O)CCCSC)NCC1(OCC)CCC1 c1(C(=O)NC2C(NC(Cn3ncc(P(C)(C)=O)c3)=O)C2)c(F)ccc2occc12 CCC1=NOC(CC(=O)NCC2CC(F)(CO)C2)C1.C1(C=O)CCC2(CC2)C1 N1(C(C(CC=CC)C)=O)CC(NC(c2c(C)nn(C(C)(C)C)c2C)=O)CC(F)C1 C1(c2nnc(-c3ccc(OC)c(Cl)c3)o2)COc2ccccc2O1 c1(CC(=O)NC(c2nocc2C(N2C(C(N)=O)CC2C)=O)C)nccn1C c1(C(=O)NC(CC)(CC)CCNC(=O)CN2CC=CC2)cc(C)cn2ccnc12 CC(C)C(C)(C)C(=O)NCC1CCCCC1NC(c1cc(Br)sn1)=O N1(C(CC2C(=O)NCC(=O)N2)=O)CC(NC(=O)Cc2ccno2)C2(CCC2)C1 CCCN=C(NC1CC(OC)C1)N1CCC(S(=O)(=O)N2CCCCC2)C1 Cc1nc(C(=O)NCC(C(C)C)NC(C2CCN(CC(C)C)CC2)=O)cc(O)n1 c1(OC)ccc2c(c1)CCC(C(N1CCC1CNC(=O)C(C)(Cl)Cl)=O)C2 c1(C(=O)NCC2C(NC(C3(C)CC=CCC3)=O)C2)cc2n(n1)CCO2 C(CN(C)N1Cc2ccccc2C1)N(CC)CC.C1(Cc2ccoc2)C(=O)N1 N1(C(C2(CC)CC2(F)F)=O)CCC(C2CC2)(NC(=O)CCc2nncn2C)C1 O=C(NN1CCCC1C(=O)NCCC1CCCCO1)C1CC2(CCC2O)C1 C(N=c1nc2sccc2c(N2CC34CCCC3(COC4)C2)[nH]1)C1(CC=C)CCCC1 c1(NC(c2c(COC)cc[nH]2)=O)ccc(NC(=O)C(=Cc2c[nH]cn2)F)c(C)c1 C(C(CNC(=O)C(c1cccc(Cl)c1Cl)(F)F)C(F)(F)F)NC(CSCC)=O c1(C(=O)NC2CCCC(CC(N3C(CSC)CCC3)=O)C2)cccc2c[nH]nc12 C1(O)(CC(=O)NC(Cc2ccccc2)C(=O)N2CCN(CCF)C2)CCOCC1 c1(C(N2CCC=C(CNC(C(C)n3cnnn3)=O)C2)=O)ccc(S(N)(=O)=O)cc1 C1(C(=O)NC(C2(C(=O)NC(c3ncc(C)o3)C)CC2)C)CC12CCOC2 c1(C(=O)NC(CC=C)CNC(=O)C(C)n2cncn2)ncc(CC)cc1C C=CCCC(c1ccccc1)NC(c1nnnn1C)(C)CC1CCCCO1 c1(N2C(CN(C(=O)CC3CCC(O)C3)C)CCC2)nc2cc(Br)cnc2s1 CCC(CC)CCCC(=O)N1CC2(CO)CC1(C(N1CC(C)CCC1C(=O)OC)=O)C2 N1(C(Cc2ccc(OC)cc2)=O)CC(NC(c2c(N)cccc2Cl)=O)C2CC2C1 Cc1cc(C)c(CC(=O)NCC2CN(C(=O)CSc3nccn3C)C3CC23)s1 c1(CNC(N2CC(F)=C(C)CC2)=O)ccc2ccncc2c1 c1(CC)c(C)[nH]c(C(=O)COc2ccccc2OCc2ccc(F)cc2)c1CC C1(C(=O)NCCNS(CC)(=O)=O)C2CC1N(C(=O)CNC(=O)C(C)(C)C)C2 N1(C(CC=CCNC(C2CCC2(F)F)=O)=O)CC(F)(F)C1C1CC1 C1(NC(c2cc(CCC)on2)=O)CN(C(C2CC3(C2)CC(O)C3)=O)CC2(CC2)C1 C1(C(=O)NC2CC(C(N(C)Cc3c(C)nsc3)=O)C2(C)C)CCC(O)CN1C Cc1cc(C)n(CC(N2CCN(C(c3cnc(O)n3C)=O)C3CC23)=O)c(=O)n1 CCCCCC(CCCCC)CC(=O)N(CC(O)CNC(=O)C1CC1)CCC C(C(C)CC(=O)N(C)CCN1CCCCCC1)NC(C(C1CC1)OC)=O C1(C(N(CCN(CC(=O)NCCCC)C)C2CC2)=O)(CC)CCOCC1 C1(C2(O)CN(C(=O)C(N3C(=O)CCC3=O)C)C2)(CNC(CC(C(C)C)C)=O)CC1 N1(C(C2N(CCC)CCCC2)=O)CC(NC(c2ncsc2C)=O)C(N=[N+]=[N-])C1 N1(C(c2cc(CCC)nn2C)=O)CCN(C(C2(Cl)CC2(F)F)=O)CC(O)C1 Cc1nc(C(=O)NCC2CCC2C(=O)NCc2csc(C)c2)co1 C(=O)(C(C)CCCC)N(C)CC1N(C(CSCCC)=O)CC(F)C1 c1(C(=O)NC2CCCC(CN(C(=O)C(N)=O)C)C2)cc2cn[nH]c2cn1 c1(C(N2CCCC(NC(C3CC4CCCCC34)=O)C2)=O)cncc2c1CCC2 C1(NC(C2(COC)CCN(C3C(C(=O)OCO)C3)C2)=O)CC2(CCC2)C1OC C1(CCC(=O)NCCCCN(C(=O)CCCc2cnn[nH]2)C2CC2)CCC(=O)C1 C1(C(C)NC(c2c(CC)nn[nH]2)=O)CCN(C(c2cn(CC3CC3)nn2)=O)CC1 C1(CN(c2nccs2)CC)CCCCN1C(c1cnc(CNC=O)nc1)=O N1(C(C2=CCCN(C(C3C(C4CC4)C3(F)F)=O)C2)=O)CC2CSCC(C2)C1 N1(CC(N2CCN(C(C(CC)(C)O)=O)CC2)=O)OC(C)(C)CC1=O Cc1cc(C(N2CC(NC(C3CC3C3(C)COC3)=O)C(CO)C2)=O)ccc1Cl c1(C(N2C3CCN(C(C4C(CC)C4)=O)CC3C2)=O)cc2c(C)cc(OC)cc2[nH]1 N12CCN(CC1)CC(N(C)C)C13COC(C1)(C3)C2=O.c1(SC)ccc(CO)cc1 Cc1cc(C(=O)NC(CNC(c2cnn(C)c2C(C)C)=O)CO)c2[nH]cnc2c1 C(CCCCC(=O)NCCCNC(c1cncc(C(F)(F)F)n1)=O)NC(N)=O C1(C(=O)NCc2c(CC)noc2)CCCCN(C(C2(Cl)CC2)=O)C1 c1(C(N(C(C)C(=O)Nc2cnc(OC)nc2)CCC)=O)cccc(C#N)c1 CC1SCCC1NC(=O)CCOCCN(C(=O)CCCn1ccnc1)C N1(C(CCCC=C)=O)CCC(NC(=O)CCOC)CC(C)(C)C1 c1(N2CCC(C)S(=O)CC2)ccc(S(=O)(=O)NCC2(C)NC(=O)NC2=O)cc1Br N1(C(c2c(CNC(C3CC=CC3)=O)n[nH]c2)=O)CCCC2(CCOC2)C1 CC(=O)CCCC(=O)NCC1CC(C)(C)CN1C(=O)CCN1C(C)CCCC1C c1(COc2ccc(C(=O)NC3CC(NC(CCCC)=O)C3)s2)ccccc1CC c1(C(=O)NC2(CCO)CN(C(c3cnccc3Cl)=O)C2)cc(F)ccc1Cl c1(C(=O)NC(CC(C)NC(=O)CCc2cccs2)C)cc2c(cc1Cl)NCC2 C(=O)(C1=CCC(NC(c2cncn2C2CC2)=O)C1)NCc1nnc(C)o1 CCCCCC(C)(CC)C(=O)N1CCN(C)C(CNC(C2CCC(C)(C)C2)=O)C1 c1(CC)ncc(C(N2CCC2CNC(c2cc(C3CC3)no2)=O)=O)c(O)n1 N1(C(Cn2cc(CNC(CC3CN(C)C3)=O)nn2)=O)CCCC2CCCC12 C#Cc1ccc(C(=O)NC(C)CNC(=O)C(c2ccc(C3CC3)cc2)O)cc1 c1(OC)ncnc(OC)c1C(=O)NCC1CCCN1C(=O)CCc1nncn1C C1(NC(C2(F)CCCOC2)=O)CCN(C(=O)CCCn2ccccc2=O)CC1 c1(C(=O)Nc2ccc(C)cn2)n[nH]c2c1CN(C(C1CC(C)(C)C1)=O)CC2 C(CC(C(=O)NCC1(CO)CCN(C)C1)NC(c1nccnc1N)=O)OCC C1(C(=O)NCCCn2cccn2)CC2CCCC2N1C(C1CC=CC(O)C1)=O C1(NC(C(C)=C(C)C)=O)CN(C(c2cc(Br)cn2C)=O)CCC1CO C1(C(=O)NCC(CC)NC(C2CC(=O)N(CC)C2)=O)CC2C(C1)C2(F)F N1(C(C(CCC)O)=O)CCC2(CCCN2C(C2(c3ccc(Br)cc3)CCC2)=O)C1 c1(OC)cc(C)c(C)cc1S(=O)(=O)N1CC2(CCC(C(=O)NC)O2)C1.S(C)(=O)(=O)N CN(CCCC(=O)N1CC(O)(CCNC(=O)CC2CCC23CCC3)C1)N=O C1(NC(c2c(C)ccs2)=O)COC2(CCCN(C(c3ccc(O)nc3)=O)C2)C1 c1(C(C(=O)NC2COC2)N(c2ccc(C)c(F)c2)C)cc(F)c(Cl)cc1Cl N1(CC=CCN=c2[nH]cnc(=N)[nH]2)CCC2(CC1)OCCC2c1nn[nH]n1 N1(C(c2c(C(C)(C)C)con2)=O)CC2(CCCCN2C(=O)CCc2ccsc2)C1 CCCC(CC)C(=O)NCC(C)N(C)C(c1cccc(CC#N)c1)=O N1(C(c2cc(C(=O)OCC)no2)=O)CC(C)N(C(=O)CC2(CO)CC2)CC1C N1(Cc2cn(CCCC=O)nn2)CCN(C(c2cnns2)C)CC1.C1CCCOC1 Cc1cccc(C(N2CC(O)CC2C)C(=O)NCc2cccc(Br)c2)n1 Cc1cc(C(N2CC(CC(=O)NCCN3CC(C)(O)C3)C(C)C2)=O)cn1C Cn1ncc(C#N)c1C(=O)NC1CC(CC(N2CCC(CO)C(O)C2)=O)C1 C(=O)(C1=CCC(C)(C)CC1)N1CC(N(C(CCS(=O)(=O)NC)=O)C)C(C)CC1 C1(CNC(CCn2cc(COCCOCCN(C)C)nn2)=O)CCS(=O)(=O)CC1 C(=O)(CC(F)(F)CC(=O)NCC1CCCCN(C(C2CCS2(=O)=O)=O)C1)OC c1(OC)cccc(F)c1CC(=O)NC1CCC1CNC(c1nc(C)ccc1C)=O C1(NC(C2CN(C(C)C)C2)=O)CC(C(=O)N(C)CCn2cnnc2)C12CCC2 C(=O)(C(O)C1CN(C(C2(C(N)=O)CC2)=O)C1)NC(c1csnn1)C c1(NC(C2(OC)CC(F)C2)=O)cc(OC)c(Cl)c(C)c1.c1(NC(=O)OCC)ccccc1 C1(CNC(CSCCC(C)C)=O)CN(C(=O)CN(C)C)CC12CC2 c1(CC)nc(Cl)[nH]c(=NCCCCNC(C2CCCCC2C2CC2)=O)c1Cl c1(CC(=O)N(C2CCN(C(CC(CC)CN(C)C)=O)C2)C)ccc2nsnc2c1 C1(C(=O)NC2(C)CN(C(C(C(C)(C)C)SC)=O)C2)CCc2ncccc2C1 N1(C(c2cccs2)=O)CCC2CN(C(=O)C=C3CCOCC3)CCC2C1 c1(CC(C(=O)N(CCCCNC(C(CC)NC(N)=O)=O)CC)C)ccccc1C CC1CN(C(C2CCC23CCC3)=O)CC1CNC(=O)CS(=O)(=O)N(C)C C1(COC)(NC(=O)Cc2cc(C3CC3)on2)CCN(C(C2CC(=O)C2)=O)CC1 C1(C(=O)NCC2N(C(c3nc(OC)c(C)s3)=O)CC(O)C2)CCOCC1(C)C c1(-n2ccc(C(N(CC(C)NC(CCC(C)SC)=O)C)=O)n2)ccc(F)cc1Cl N1(C(CCc2n(C)ncn2)=O)C2CC=C(C(=O)NCC(O)CO)C1CC2 c1(OC)ccc(NC(=O)CC(=O)NCC2CN(C(c3nncs3)=O)CCO2)cc1 c1(C(=O)NC2CCCN(C(=O)CC3CCC3)CC2F)n[nH]c2ccc(Br)cc12 C1(NC(c2nn(CC)nc2C)=O)C2CCCN(C(C3CC3C#N)=O)C2C1(C)C C1(C(=O)NC(c2ccoc2)C)CCC(NC(C2CCCS2)=O)C1 c1(CC(=O)NCC(CO)NC(c2nc(C(C)C)sc2)=O)cccc(Cl)c1F c1(C(=O)NC(C2(O)CCN(C(c3n(C=C)ncc3)=O)C2)C)cc2c(nn1)CCC2 N1(C(COCCN(C)C)=O)CC(O)CC1CNC(c1nncn1C1CC1)=O N1(C(C(c2cn(C)nc2)O)=O)C2CCC1C(C(=O)NC1CCC3(CCC3)C1)C2 CCCCCC(C)(C)C(=O)NC1CN(C(=O)C(C)(CC)CC)CCC1CO c1(C(=O)NC)cc2c(F)ccc(Br)c2[nH]1.CC(C)CC(=O)C(N1CCCC1CN)=O c1(OC)cc(I)ccc1COC(=O)C(C)(C)C1(N(C)C)CCCC1 CC1CCC(NC(=O)CNC(c2ccccn2)=O)CN1C(=O)CC1CC1C C(C(CCC)C(=O)N(CC(C(C)C)OC)C)NC(c1n(C=C)nnc1)=O c1(NCC2CCN(C(C=Cc3cncc(OC)c3)=O)C2)ccc([N+](=O)[O-])nc1 CCC(CC)(CC)C(=O)N1CCOC(CN(C(=O)Cc2ccc(SC)cc2)C)C1 C12(C(N(C3CN(C(CS(N)(=O)=O)=O)CC3O)C)=O)C3C4C1C1C2C3C41CO c1(C2CN(CC(c3ccc(O)cc3)(C)O)C2)ccccc1F c1(CC(N2CC(CCCCNC(C3C(C)(C(C)C)C3)=O)C2)=O)c(O)ncnc1O N1(C(C2CC(CCNC(C(C)F)=O)C2)=O)CCC(C(=O)O)(C(C)C)C1 c1(C(=O)NCC2(NC(C3CCOC(C)C3)=O)CC(OC)C2)cnc(O)n(C)c1=O Cc1cccc2[nH]cc(C(=O)NCC(C)N(C)C(c3csc(Cl)c3Cl)=O)c12 C(CCNC(=O)CC(C)F)(C(C)C)NC(C(CC)Oc1ccccc1)=O c1(C(=O)NC2CC(=O)NC2)nc(O)nc(O)c1[N+](=O)[O-] C(=O)(C(C)CC(C)C)N1CC(C(C(=O)NCC2CCCC2(C)C)OC)C1 Cc1cnc2cc(C(=O)NC3CC(C)(NC(=O)CC4CC5CC5C4)C3)nn2c1 CC1(C(=O)NCC(N2CCN(C(c3noc(C(N)=O)n3)=O)CC2)=O)CCCOC1 C1(CNC(CCN(C)CC)=O)CN(C(=O)CCc2ccco2)CC12CCC2 c1(C(=O)NC(CCC)C(=O)N2CC(CO)C(O)C2)cc(C)c(N)cn1 C1(C)(NC(=O)NC(c2cc(C(F)(F)F)ncc2F)C)CC(O)CN1C c1(OC)ccnc(C(=O)NCC2CCCCN2C(C2CC(C(C)C)C2)=O)c1 C=CC(C)CCNC(=O)CN(C(=O)C(C)n1cccn1)CCC N1(C(CC(CCC)C2CC2)=O)CCC(O)C(O)(C(=O)NC(=O)NN(C)C)C1 c1(C(N(C)CC2(NC(C3CC3C(C)(C)C)=O)CC2)=O)ccc2nc(Cl)nn2c1 c1(C(C)NC(=O)C(N2CCC(c3cnccn3)CC2)=O)ccnc(Cl)c1F c1(Cc2onc(C(c3ccc(Br)cc3)C(=O)OC)n2)cc(C)ccc1C(F)(F)F N1(C(CC2(C)CC2)=O)CC(O)(CNC(c2cnn(-c3ccccc3)n2)=O)C1 c1(N(CC)CC)ccc(NC(C2CC(O)CN2Cc2ccnn2CCF)=O)cc1 N1(C(CS(CCCC)(=O)=O)=O)CC2(CCC(NC(=O)CCCN(C)N=O)CC2)C1 c1(C(=O)NCC(C2CCCC2)NC(C2(O)CCC2)=O)cnc2c(c1)CCCO2 C1(C(=O)OC)CN(C(C2(C#N)CC3CC3C2)=O)CC12CCCCCC2(F)F c1(OCC(=O)NCC(CN(C)C(C2CCC2C(F)F)=O)O)ccccc1F C#CCC(C)(CC)C(=O)NC1CCN(C(c2cnn(CC(C)C)c2C)=O)CC1 C1(CC=C)(C(=O)N(CC(O)COC)C)CCCN1C(=O)Cn1cc(CO)nn1 CN(CCCC(=O)N1CC(CNC(c2cnn3ccsc23)=O)CC(C)(C)C1)N=O c1(CC)cnoc1C(=O)NC(Cn1cncn1)C(=O)N(CCC(F)(F)F)CC CC1CCC=C1C(=O)NC1CCN(C(c2ccc(Br)cc2)=O)C1C S1(=O)(=O)c2ccccc2NN(C)C(C)CN1.C(C)(C)(C)OC(=O)NCC C1(NCC(c2ccc(F)cc2)N(C)C)CC(F)(F)C1(C)C c1(-c2nc(CCCCC)nn2C2CC=CC2)cc(Cl)cc(F)c1Cl C1(NC(C(F)=CC)=O)CN(C(C2(NC(=O)NC)CCCC2)=O)CC1C c1(COC)cnc(OC)c(C(=O)NC(c2ccc(Cl)cc2)C(C)C)c1 C(c1ccccc1CN1CCN(c2ncncc2C#N)C2CC12)=CC(=O)O N1(C(c2cnc(C(C)=O)s2)=O)CC(C)N(C(=O)CC2=CCCCC2)CC1C C(CNC(c1ccc(C(C)=O)[nH]1)=O)(CC(=O)N(CCC(O)CO)C)OC C1(CCC(=O)N(CCCCN(C(C(C)SCC)=O)C)C)NC(=O)NC1=O C(C(C(=O)N1CCC1(C)C(N)=O)NC(=O)C(O)Cn1cncn1)OC(C)C C12CCCN(C1)C(=O)C1(CC1)COC(C)C(=O)N2C.C(COC)OC C1(CNC(C=COCC)=O)(COC)CCCN1C(C1CC(=O)N(CC(C)C)C1)=O Cc1ccc(I)c(NC(C2CCCC2NCc2ccc(Cl)cc2F)=O)n1 N1(Cc2ccc(CC=C)cc2F)CC(C2CC2(F)F)C1 N1(C(c2ccc(F)c(Br)c2)=O)CC2CN(S(=O)(=O)c3cn[nH]c3)CC2C1 C(CC1=CCCCC1)NC(C1C2CC3C(C2NC(C24COCC2C4)=O)C13)=O n1(CC#C)cnnc1C(=O)NC1CC(O)(CNC(C2CNC(=O)N2)=O)C1 Cc1cccc(Cl)c1N(CC(=O)NCCCCCN(C(=O)C=CCO)C)C C#Cc1cccc(C(=O)NCCCCC(C)NC(C2CC2C)=O)c1C C(=O)(C#CC1CCOC1)N1CCN(C(c2cc(C)c(C)s2)=O)CC1C N1(C(=O)C[SH](C2CCC2)C2CC2)CCC(C(F)(F)F)CC1.N1(CC)CCOCCC1 C1(C)(C(=O)NC(CC2CN(C(CC(=C)Br)=O)C2)C)CCN(C)C1=O N1(C(C(CC)O)=O)CCC(C)(CNC(c2cc(Br)ccn2)=O)C1 c1(OC)cc(NC(=O)C(N2CCC(C3CCC(C(F)(F)F)O3)CC2)=O)n(C)n1 C(=O)(C1=CCCOC1)NC(CCNC(CN(C)CC)=O)C N1(CC(=O)C(=O)Nc2ccccc2)CCC2(CC1)COCCC2N.C1(=O)CN1C c1(C(=O)NCC2(C(C)(C)O)CN(C(CSCCOC)=O)C2)cnc2c(c1)COC2 N1(C(C(C)(C)NC(=O)NCc2ccc(C3CC3)o2)=O)CCc2ccccc2C1 CCCC(C)(CCC)C(=O)NCCCC(C1CC1)OC.c12coc(n1)COC2=O O=C(CC(F)(F)C(F)F)NCCCCNC(c1ccn(C2CCC2)n1)=O C(=O)(N=c1nc[nH]n2cncc12)N1CCC(C)C(F)(F)CC1 Cc1ccccc1CCCNC(c1ccc(-c2cnc(=N)[nH]c2)nc1)=O C#Cc1ccc(Cl)c(C(=O)NCC(C)(C)CN(C)C(c2nscc2C)=O)c1 N1(C(C2N(C(c3cc(C)nn3C)=O)C3C(C2)C3)=O)CCc2cnn(C)c2C1 C12(NC(C3CC4CCC4C3)=O)CCC(C1)N(C(c1ccc(Br)o1)=O)C2 c1(C(=O)NC2CCCC2NC(C2CCCCO2)=O)ncc(F)cc1F c1(C(N2CCCC(C(N(C)C3CC3)=O)C2)=O)cc(F)cc2nn(C)cc12 Cc1ccc(C(N2CCC(NC(c3ncn(C)n3)=O)C(F)C2)=O)cc1[N+](=O)[O-] Cn1ccnc1CCC(=O)NC1CCC1CNC(C1CSCCS1)=O C=C(CNC(c1cncnc1)c1ccccc1)C(C)C N1(C(=O)NC(c2ccc(C#N)cn2)C)CCC(P(C)(C)=O)CC1 C1(C(N(C2CCCO2)CC)=O)CCCN(C(=O)CCN(C)CCOC)C1 c1(C(C(=O)NCC(CNC(c2cccc(C(C)=O)c2)=O)OC)C)cccc(C)c1 CC(C)CC(CC(=O)NC1CN(C(C2CCN(C3CC3)C2)=O)C1)CC(N)=O C1(CN(C(COC)=O)C)CCCCN1C(c1cc(C)n(-c2ccccc2F)n1)=O Cn1cnc2c(N3CCC3C(N3CC4(CC4)CC3C)=O)ncnc12.C(C)(C)(C)O Cc1cn2c(n1)CC(C(N1CCCC(NC(=O)C(c3ccc(C)o3)C)C1C)=O)C2 C(CCC(=O)N1CCC1CN(C)C)N(C)C(C1C=CCS1)=O C(C(O)CN=c1ccnc(C(F)(F)F)[nH]1)NC(C(c1ccc(F)cc1)C)=O Cc1cnc(C)c(NC(=O)CC2CC3(C2)CN(C(=O)CC2CCCCC2)C3)c1 C12(N(C)C(c3csc(Cl)c3)=O)CCCC1CN(C(=O)C=Cc1cnn(C)c1)CC2 N1(C(C(CC=C)NC(C)=O)=O)CCC(COC)(NC(c2csc(=N)[nH]2)=O)CC1 CC1(NC(C2CNC(=O)N2)=O)CC(NC(c2ccncn2)=O)C1 CON(CCC(=O)N1CCN(C(=O)C(C)(C)C#N)CC1C)C(=O)C1CC1C N1(C(C(CCC)(F)F)=O)CCC(C(N2CC(C3CC3)(OC)C2)=O)CC1(C)C C(=O)(C1=CNC2=NCCCN12)NCC1N(C(CC(C=C)CC)=O)CCCC1 c1(C(=O)NCC2OCCCN(C(C(CC)OCC)=O)C2)csc2ccncc12 N1(C(CCN(CC(N2CCCCC2)C)CC)=O)CC(NC(=O)OC(C)(C)C)C(C)C1 n1(CC)nc(C(N2CCC2CC(=O)NCC=CBr)=O)c(C)n1 C(CCC(=O)NCC(C)C(=O)NC1CCN(CCCF)C1)OCCC c1(NCC2CCC(N(C)C)CC2)nccc(=NC2C3CCCC23)[nH]1 C1(OC)CCN(C(C2CCN(C(=O)C3=COCC3)C2C(C)C)=O)C1C c1(OC)ccc(C(N2CCCC2CCNC(C2(CF)CC2)=O)=O)nc1 C1(C)(C(=O)NCC(CC)n2cccn2)CC(O)CN1C(c1n[nH]c(=N)[nH]1)=O C1(NCc2cc(C(=O)OC)no2)CC12CC(NC(=O)CN1CCCC1C)C2 C(C(CC(F)(F)F)NC(=O)C(O)c1ccco1)NC(C(C)(C)N(C)C)=O Cc1cn2c(n1)C(C(=O)NC(C)(C)CN(C)C(c1cnc(O)c(C)c1)=O)CCC2 C(C(C)(CC(C)C)NC(=O)Cc1cc(C2CC2)no1)NC(CCC(C)OC)=O C1(C(=O)N(C)CCN(C(=O)CN2CCC(C)C2)C(C)C)(OC)CCOCC1 Nc1cc(C(N2CCCCC2CNC(=O)CC(C2CC2)C2CC2)=O)cc(Cl)n1 C1(CC(=O)NC(C2CN(C(=O)COc3ccc(CO)cc3)C2)C)COCCOC1 c1(CC(=O)NCCN(C(=O)CC2(CO)CC2)CCC)ncsc1Br N1(C(C(C(C)NC(c2cc(CC)no2)=O)(C)C)=O)CCOCC(C)(C)C1 N1(C(c2cc(N(C)C)ncc2)=O)CCCC2(NC(c3ccccc3F)=O)CC2C1 C#CCCCCCC(=O)N(CC(O)CN(C(=O)C(F)(F)C(C)(C)O)C)C n1(CCC)nnnc1C(c1nc(C)cs1)NCCC(C1CCOCC1)O Cn1cnc2cc(C(N3CCCC(CCCO)C3)=O)cnc12 N(C(=NCC(=O)NCC(F)F)NC1CCOCC1)CC(c1ccccn1)C C=C(C)C(C)(O)C(=O)NCCCCCCN(C(=O)Cn1cncc1C)C CN1CCC(CO)(CNC(C2(C)CCCN2C(=O)CC2CNC(=O)O2)=O)C1 N1(C(C(=O)N(CCC2CCN(C(CC)C)C2)CCN2CCCC2)=O)CCC(C)CC1 c1(CC)nc(C)c(C(N2CC(NC(=O)C=C3CCOCC3)C(C)C2)=O)o1 C(N=c1nc2c(c[nH]1)COCC2)C1(CCNC(C2C(C)(C(C)C)C2)=O)CC1 Cc1cccnc1C(N1CC(NC(=O)Cc2ccc(CN(C)C)cc2)C2CC12)=O C1(C(C)(C)C)CC(C(=O)NCC(C2CC2)NC(c2ccc(N)cc2O)=O)=NO1 c1(CNC(C(CSC)OC)=O)cccc2c1OC(F)(F)O2 N1(C(c2cccc(SC)c2)=O)CCC(NC(c2cc(F)n(C)n2)=O)CC1C c1(NC(c2ccc(C(C)=O)cc2)=O)ccc2c(c1)CCC(C)(C)O2 c1(C(=O)NCC2CCC(NC(CC(C)O)=O)CC2)cnc2cc(Cl)ccn12 CCC1C(=O)N1.c1(C(N(CC(C)C(=O)OC(C)(C)C)C)=O)c[nH]nc1C(F)F c12cn(cn1)CC(=O)NCCN(C1CC1)C2=O.C1(NC(C)=O)CC(CC#N)C1 C=CC(CCC)CC(=O)N1CCC(C)C(CC(=O)NCCCn2cncn2)C1 c1(CNC(=NCCSC)NCC2COCC(C)(C)O2)c[nH]c2cnc(Cl)cc12 c1(C)cccc(C#N)c1.C(C(=O)NC)(C(C1CCCCC1)NC)NC1CC1 c1(N2CCC(C)(NC(=O)CN3C(=O)NC(C)(C)C3=O)C2)nc(Cl)ncc1[N+](=O)[O-] C1(C)(C(=O)NCC(C)(C)CNC(C2CC(n3ccnn3)C2)=O)CCNC(=O)C1 C(CS(=O)(=O)C1CCOCC1)NC(C1CCC2C3CCC(C3)C12)=O CC(C)(O)CCC(=O)N1CC(CNC(c2cc(C3CC3)no2)=O)C(C(F)(F)F)C1 N1(C(CCSC)=O)CCN(C(=O)CC2COCCO2)C2COCC12 N1(C(=O)CCc2ccco2)CC2CCC(C1)N2C(c1ccc(O)cn1)=O C(=O)(NN1CCCCCC1=O)C1OCC(CC(=O)OC)C1 CC(C)(C)C(CNC(=O)CC(C)(O)C1CC1)NC(C1CC(c2ccccc2)C1)=O N1(C(CC(C)(C)O)=O)CCCCC(C2CN(C(=O)CC3CCC(F)(F)CC3)C2)C1 CCC(COC)C(=O)N(CCCCO)Cc1ccc(CNC(c2cnc(Cl)s2)=O)cc1 c1(OC)ncnc(OC2(C(=O)NCCNC(=O)COCCF)CC2)c1F c1(C(N2CC3CC3(C(=O)Nc3cc(F)c(Cl)c(Cl)c3)C2)=O)ccc(Cl)c(Cl)c1Cl c1(C(=O)OC)cc(C)cnc1NC1CC(NC(=O)Cn2nccn2)C1 C12(NC(Cc3c(C(=O)OC)cccc3)=O)CCN(C(=O)CCC(C)C)CC1C2 c1(OC)ccc([N+](=O)[O-])cc1C(=O)NC(C)CCNC(c1conc1C(C)C)=O c1(C(N2CC3C(CNC(=O)C4=CCC4)C3C2)=O)cc(F)c(Br)cc1F N1(C(c2c(C)[nH]cc2)=O)CCN(CC(=O)NC(C)(CO)C2CCCC2)CC1 c1(C(N(CCOC)CCNC(C23CC(F)C2C3)=O)=O)cc2ccsc2n1C CCC(C(=O)NCc1ncoc1C1CN(C(=O)COCCCOC)C1)C(C)O N1(C(CCc2cnc(C)o2)=O)C2CCC1CC(CNC(=O)C1=C(Cl)CCC1)C2 c1(C(N2CCC(NC(=O)CCCn3cncn3)C2)=O)cccnc1Br N1(C(c2cnn(-c3ccccc3)c2)C(=O)NCC)CCC(O)(c2ccccc2)C1 C=CCCCCCC(=O)N1CCC(NC(C2CC3OC2C2CC32)=O)C12CCC2 Cc1nc(O)ccc1C(=O)NC1CCCCC1CNC(=O)C=Cc1csnc1C N1(C(CCCC#C)=O)CCN(C(=O)CC2CCN(C)C2=O)CC12CCC2 C1(CC(N2CC(C)C(O)C2)=O)CCCCC12NC(=O)NC2=O N1(C(C(C)CCO)=O)CCCC(NC(C2CCCC2C)=O)CC1 C(=O)(C#CC1CCCCC1)NCC#CCOCCc1cc(C(=O)OC)no1 C1(F)(CNC(C(CC)SC)=O)CCC(CNC(c2ccnnc2)=O)CC1 N1(CCC)CCC(N=c2nc3scnc3c(NCCCc3ccccc3)[nH]2)CC1 c1(C(=O)NC(C2CCCN(C(c3cnsn3)=O)C2)C)ccc2nnc(Cl)n2c1 N1(C(C(C2CCCC2)NC(c2cc(C)nc(C)n2)=O)=O)CCCCN(C)CC1 S(=O)(=O)(c1ccc(Cl)cc1)NCCC(=O)NCc1c(OC)cc(F)cc1 CCCC(C(=O)NCCC(=O)NCC(=O)Nc1cccc(F)c1)N(C)C C1(SC)CC(c2nnnn2C(C)(C)CC)(NCCOC2CCOC2)C1 c1(C(N2C(CNC(c3ncc(C)c(Cl)c3)=O)C(C)CC2)=O)ccc2c(c1)CCC2 c1(OC(C)C)cccnc1C(=O)NC(C1CCCCC1)CNC(=O)C=C(Cl)Cl CC1CCC(C(=O)NC2C3CCC(C3)C2C(N)=O)N(C(c2ccccc2)=O)C1 C(c1ccc(F)cc1F)=CC(=O)NC(C)CCCNC(c1c(Cl)csc1Cl)=O c1(OC)cc(CC(=O)NC2CCCCC2CO)nc(NC2CSC2)n1 N1(C(Cc2cc(C)ncc2)=O)CC2(C1)CN(C(c1cnccc1Cl)=O)CC2CO Cc1cc(N2CCCC(CCNC(c3cc(Cl)cs3)=O)C2)ccc1[N+](=O)[O-] CCCC(C(=O)OC)C(=O)N1CCC(C)(C)C(NC(=O)Cn2cncn2)C1 C1(COC)CC(CNC(c2ccncc2F)=O)N(C(c2cnc(C(C)=O)s2)=O)C1 N1(C(C2(CCC)CCC2)=O)CC(CNC(c2ccc[n+]([O-])c2)=O)C(O)C1 N=c1[nH]c2c(s1)CCCC2C(=O)NC1CCCCC1CNC(=O)Cc1cncs1 C1(C(CCC)C)CCCN1C(=O)COCCNC(=O)C(C1CC1)SC N1(C(C2N(C(c3cncc(C=C)c3)=O)CCOCC2)=O)CCCC(C)(CC)CC1 N1(C(Cc2c(C)cnn2C)=O)CCC(NC(C23CCC(CO)(CC2)C3)=O)CC1C c1(NC(=O)C(c2ccc(Cl)cc2)=O)cccc(NC(c2cc(Cl)cs2)=O)c1 c1(C(=O)NC(C(C)NC(c2cnc(C)[nH]2)=O)CO)c(C)ccc(F)c1O c1(SC)ccc(NC(=O)CN2CCC(N(C(=O)C(n3ccnc3C)C)C)C2)cc1 N1(C(c2n(CC)ncc2Cl)=O)CC(NC(=O)CCCC(=O)OC)C(C)(C)C1 C1(NC(CC)=O)CC(CO)N(C(=O)C(C)CC)C1.C(=O)(C=CC(C)C)N c1(C(=O)NCC(C)C(=O)N(CC(C)(C)O)C)cccc2ccoc12 O=C1Cc2c(C(=O)NC3CCN(Cc4cccc5ncccc45)C3)cccc2N1 N1(C(C(CC)OC)=O)CCC(CNC(C2(OCC)CCC2)=O)C(F)(F)CC1 [N-]=[N+]=NCCCC(=O)NCCOCCCNC(c1ocnc1C1CC1)=O c1(C2(C(=O)NCCCN(C(C(CC)SC)=O)C3CC3)CC2)ccc(Cl)nc1 c1(C(=O)NC2(CC=C)CCN(C(=O)CN(C)C(N)=O)C2)ccc(F)c(F)c1 C(CO)(CC(F)F)NC(=O)CCOC1CCCCC1 c1(C(N(CC(CC)NC(=O)CCF)C)=O)c[nH]c2cc(F)cc(F)c2c1=O c1(C(=O)NCC(CC)(CC)NC(C2CC2C2CC2)=O)cncc(F)c1C N1(C(c2n(C)ccc2)=O)CCC2(C1)CN(C(=O)C=Cc1n[nH]c(=N)s1)C2 CCC(O)C(F)(F)C(=O)NCCCN(CCCNC(=O)CC(F)(F)F)C C1(NC(c2ccc(C)nc2)=O)CC(C)CN(C(c2sccc2Cl)=O)C1 n1(CC)nnc2c1CCC(C(=O)NC1CC(C)N(C(c3csc(C)c3C)=O)C1)C2 N1(C(Cc2c(C)n[nH]c2C)=O)CCN(C(c2ccn(C)c2C)=O)CC(O)C1 C1(CNC(CSc2onc(C)n2)=O)C(C)CCCN1C(=O)C1=CCOC1 CC#CCC(C(=O)N1CCC(OC2CC2)C1)NC(C1CCC2CC12)=O C1(NC(C=C(CC)C)=O)CCC1NC(=O)C(=O)NC(C)C N1(C(C2N(C(c3cc(OC)ncn3)=O)CCC(F)C2)=O)CC2CCC(C1)C(=O)N2 CCCC(=O)N(CC(=O)N(CC(O)CO)C)C1CC1.C1C(=O)N1 N1(C(C2N(C(CCC)=O)CSC2)=O)C2CCC1C(NC(c1cc(Cl)no1)=O)C2 C1(NC(C2CC(N(C)CC)C2)=O)CCCCCN(C(=O)CN2CC(C)(OC)C2)C1 c1(NC2C(CC(=O)NC3CCN(C(C)=O)CC3)CCC2)cnc(Cl)cn1 CCCCC(C)C(=O)NC1CCCCC1CNC(=O)C(C)=CC1CC1 CP(C)(=O)C(O)C(=O)NCCC(c1cccs1)NC(C1(CC2CC2)CC1)=O c1(OC)cc(C(c2nnnn2CC(F)F)NCC(CCSC)OC)cc(F)c1 C1(NC(CCNC(C)=O)=O)CC2(CCN(C(C3CC(C)CC(C)(C)C3)=O)CC2)C1 c1(C(=O)NCc2occ(C(=O)NC3CC(C(C)=O)C3(C)C)n2)cnn2c1CCC2 c1(OC)ccc(C)cc1C(N1CCC(NC(=O)CNc2ccccc2)C(O)C1)=O c1(C(N(C)CC2C(NC(C(F)=C(C)C)=O)CCC2)=O)nccc(C)n1 C1(NC(=O)CCCn2ccnn2)CCCC12CCN(C(c1ncncc1Cl)=O)C2 C(=O)(C1=CS(=O)CCC1)NCC1(O)CCN(C(C(C)(C)c2cccs2)=O)C1 CC1CCN(CCC2CCC(OC(C)(C)C)CC2)C1(C)C n1(CC)nc(C(N2CCCC(CCNC(=O)CCNS(=O)(=O)CC)C2)=O)cc1C c1(CC(=O)NCC2(C)CCN(C(C(C)S(N)(=O)=O)=O)C2)c(F)cc(F)cc1F C(c1ccc(F)cc1F)=CC(=O)NCCN(C(c1nc(C)ccc1F)=O)CC Cc1cn(CC(=O)N(C2CCN(Cc3cccc4c3OCO4)C2)C)c(=O)nc1O c1(CC(=O)NCC2(F)CC(NC(c3scc(C)c3Cl)=O)C2)cccc(F)c1F c1(C(N(C(C)CNC(=O)CC2CCCC2O)C)=O)cn(C)nc1C(F)F C1(NC(Cc2ccc(C)o2)=O)CN(C(c2cc(-n3cnnc3)ccn2)=O)C2CC12 c1(N2CC(C)(COC)OCC2)nc(=NCc2n[nH]cc2Br)[nH]c2c1CC(C)CC2 N1(C(C23CC(C)(C2)C3)=O)CCC2CN(C(C3CCC(F)(F)C3)=O)CC2CC1 c1(-n2cc(C(=O)NCCc3ncc(C(C)(C)C)s3)nn2)ccccc1Cl c1(CN(c2nc(C3CCC3)no2)C(C)C)cccc(OC(F)(F)F)c1 Cc1nnc2n1CC(C(N1CCCN(C(=O)C(C)NC(N)=O)C(C)C1)=O)C2 c1(CNC(COCC(C)(C)C)=O)ccc(CNC(c2sccc2F)=O)cc1F C12(NC(=O)CCc3ncc[nH]3)CCN(C(c3cnc(SC(F)(F)F)s3)=O)CC1C2 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(C)Cc2cccnc2)C1(C)C O=S(=O)(c1cc(Cl)cc2cccnc12)N1CCc2nnc(-c3ccsc3)cc2C1 C(=O)(N=c1[nH][nH]cc1Br)N1C(c2cccs2)CC1=O.c1(OC)cccc(C)n1 c1(C(=O)NC2C(OC)CN(C(=O)CC3CCCO3)C2)cn2c(n1)CCC2 N1(C(COCCCOC)=O)CCCC(C)C1CNC(c1ocnc1C)=O Cc1nn(C2CCOC2)cc1C(N1CCC(NC(c2ccccc2CO)=O)C1)=O N1(C(C23N(C(CC4CC(=C)C4)=O)CCC2C3)=O)CCCC2(CCCC2)C1 c1(C(N2CCC(Oc3ccccn3)C2)=O)cc2c(nc1O)CCCC2 c1(NCC2(OC)CCC2)ccc(S(=O)(=O)NC(c2ccc(CF)cc2)C)cc1Cl C(=O)(C1CCCc2c[nH]nc21)N1CCC2(C(NC(C3CC4(CSC4)C3)=O)C2)CC1 C(=O)(C1=C(Cl)CCOC1)N1CCC(N2CCN(C(C3(C)CC(C)OCC3)=O)CC2)C1 N1(C(CC(C(C)C)C)=O)CCCC2(CNC(c3ccoc3)=O)CCCC12 C#CCC(C)(CC)C(=O)NCC1CCCN(C(=O)CCCS(C)(=O)=O)CC1 c1(CN(C(C(C)OCC)=O)C)nc(-n2cccn2)cs1 C#CCCCC(C)C(=O)NC1(C2CN(C(c3csc(-c4ccoc4)n3)=O)C2)CC1 CN1CC2CCC1CN2C(C1(F)CCN(Cc2c(F)ccc(Cl)c2Cl)C1)=O C=CCCCCCC(=O)NCCCC1(NC(=O)Cn2c(C)csc2=O)CC1 CC(O)C(C(=O)N1CC(CNC(=O)C(c2ccc(Cl)cc2)(C)O)C1)N(C)C c1(CC)nc(C(=O)NC(C2CCN(C(=O)CCCCSC)CC2)CO)c(N)s1 c1(SCC(=O)N(C)CC2CCN(C(C(CC)O)=O)C2)ccc(C)cc1C Cc1cc(C)c(C(=O)NCC2CN(C(=O)C=CC3CCCN3C)CCCO2)cn1 C1(CCN(C(C2C(C)CCC2)=O)C)CCCCN1C(=O)C=CCN1CCOCC1 C1(CNC(CC)=O)CC2COCC2N1C(c1ccc(OCC(N)=O)cc1)=O c1(NC)cnnc(C(=O)NCC2CC(NC(C3CCCN3C3CCCC3)=O)C2)c1 N1(C(C(CC)N(CC)CC)=O)CCC2C(CCN2C(=O)CNS(=O)(=O)CC)C1 N1(C(C=C(CC)C)=O)CCC(CCCNC(=O)C=Cc2ccsc2C(F)F)CC1 Cc1ccc(C(=O)NCC(C(C)(C)C)NC(C2CCCC2)=O)c(Cl)c1 C1(c2cn(CCCCF)nn2)(NC(C2CCN(CC(F)F)C2)=O)CC2CCC1CC2 C#CC1CCCN(C(=O)C(CCC=C)NC(=O)C(C)Cn2ccnc2)CC1 c1(-c2n(C(C=C)C)nc(C3CC3)n2)cccc(S(=O)(=O)CC)c1 CS(=O)CNC(=O)CCC1CC1CSC1CC1.C12(CCC1)CC(=O)N2 C(N=c1nc2c(ncn2CC)c(N(C)CC2COCCO2)[nH]1)c1c(CC)c[nH]n1 C(CC(CC)C(=O)N1CC2CC(NC(C3CC4CCC(C3)C4)=O)C2C1)=CC Cn1cc(C(N2CCC2CNC(=O)C(F)C2CC2)=O)nn1 Cc1n[nH]c(C)c1CNC(=O)C(c1ccoc1)NC(C1CC(C)CCO1)=O N1(C(c2cn(CC)nc2C)=O)CCC(C2CC(NC(C3CC(C)(C)C3)=O)C2)C1 Cc1nc(CC(N2CCC(CN(C(=O)CCC3CCC(C)O3)C)C2)=O)cs1 c1(NC(COC)CCOC)ncnc(N2CCCC(C(N)=O)C2)c1C c1(C(CC)NCCCC2CCOCC2)ccc(F)cc1 C(CC)(C(=O)NCCNC(=O)C(C)C1CC(NC(=O)OC(C)(C)C)C1)NC C1(NCc2cn(CC)nc2)CN(C(=O)CC2CCCC2)CC1O N1(CC)CCCC(CNC(=O)C(O)CNC(=O)Cc2ccc(O)cc2)C1 Cc1cc(C(N2CCCC(C)(C(=O)NC3COCC3O)C2)=O)c(F)cc1Br c1(NC(C2CN(c3ccc(C#N)cc3)C(=O)C2)=O)ccc2nc(F)ccc2c1 c1(C(C=C)N(CCCF)C)cc(OC(C)C)c(OC)c(OC)c1 CC(=O)CCCC(C)C(=O)N1CCCC1C(=O)N(CC(=O)N(C)C)C Cn1nnnc1C(CNCCCc1ccc(Cl)s1)C(=O)OC(C)(C)C N1(C(CNC(=O)OC)=O)CC(OC)OCC1C1CC1.C12(CCCO1)C(=O)NC2 c12cc([nH]n1)CNC2=O.C1(CCNC(=O)CC2CC2)(N(C)C)CCC1 C(=O)(C(CCC(N)=O)N(C)C)N1C(CNC(c2cc(CC)c(C)s2)=O)CCC1 Cc1c(CNC(=O)CC(c2ccc(F)cc2)N)nc2ccccn12 c1(COCC(=O)NCC(C(C)C)(C)NC(C2CCCO2)=O)ccc(F)cc1O c1(C(=O)NC2CCCC(N(C(c3c(OC)nccn3)=O)C)C2)c(C)nn(C)c1C Cc1nc(CCC(=O)NC2CN(C3CCCCC3)C2)sc1C Cc1cn(C)c2nc(N3CCOC(CC(=O)Nc4ccc(Br)nc4F)C3)ncc12 C(CC(C)C)(C(=O)N(C)CC1(O)CN(C(c2cncc(C)n2)=O)C1)OC N1(C(C=CC)=O)C2CCC1CN(C(=O)CC1OCCC1(C)C)C2 c1(C(N2C(C(=O)NC(c3ccccc3)CC=C)CCC2)=O)cnc(C(N)=O)cn1 C1(C(N(CCOCC)CC)=O)CCN1C(=O)Cn1nccn1 N1(C(c2[nH]c(=NCC)sc2)=O)CCC2(CC1)OCCc1sc(C(=O)O)cc12 C1(CCNC(C2(OC)CC2)=O)C(C)CCCN1C(=O)CN1CCCCCC1=O C#Cc1ccnc(C(=O)NCC2CCC(C)CN2C(c2ccc(SC)cc2)=O)c1 c1(C(=O)NCC#CCNC(=O)COCCc2ccccc2)cc(F)cnc1O C1(CNC(=O)CCn2ccnn2)CC2CCC(C1)N2C(c1cc2sccc2[nH]1)=O C1(F)(CNC(CCOCCC)=O)CC2CCC(C1)N2C(=O)C(CC)C(F)(F)F c1(C(N2CCN(C(c3n(CC)ncn3)=O)C(CO)C2)=O)ccc2c(c1)N(C)CC2 C(C)(CCC(C)(C)C)NCCCNS(c1c(OCC)ccs1)(=O)=O CCC(CNC(=O)C(O)C1CCCC1)N(C(=O)C(C)OC1CCCC1)C C1(C(=O)NC2CC2C2CC2)CC2CCC(C1)N2C(c1cc2ccccc2[nH]1)=O C1(C(C)C)C(C(=O)NCc2ccnn2C)CCN1C(=O)CN1CCNC1=O c1(C(=O)NC(C)CN(C)C(C2(CCF)CC2)=O)cc(=O)c2ccc(O)cc2o1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCCN(C(c1cnc(CO)nc1C)=O)CC C1(C)(OC)CCN(CC=C2CCN(C(c3cnc(C4CC4(F)F)s3)=O)CC2)CC1 N1(C(C2CC(C)(O)C2)=O)CCC(F)C(NC(=O)C(F)CNC(=O)OC(C)(C)C)C1 n1(C(C)C)nc(C2CCOC2)nc1C1CC(=O)N(C)C1 N1(CC(=O)N(CCC)CCC)CCC(C(C)(C)CNc2sc(C)cc2Cl)CC1 Cc1ccc(F)c(OC2CCN(c3nc(C(=O)O)nc(=N)[nH]3)CC2)c1 C(C(C)(C)C(=O)NCC(C)(C)CNC(c1cc(C2CC2)[nH]c1C1CC1)=O)OC N1(C(COCCC)=O)CC2CN(c3ncc(Br)c(C(F)(F)F)n3)CC2C1 c1(SC)cnn(C)c1C(=O)NC(C1CCOC1)CNC(=O)CN1CCCCCC1 O(NC(=O)C(C(C)(C)C)n1cc(CS(C)(=O)=O)nn1)CC(CC)C c1(C(=O)NCCC2OCCN(C(C(C=C)O)=O)C2)ccc(F)c(Cl)c1 c1(C(=O)NCC(C)(C)CNC(=O)Cc2cc[nH]n2)ccc2n[nH]cc2n1 Cc1occc1CNC(=O)C(c1cccs1)NC(=O)C(C)N(C)C CCCC(C)CC(=O)N1CC(CCCCNC(c2ccoc2C2CC2)=O)C1 c1(C(N2CCC(C(=O)NC3CCN(CC)C3=O)C2)=O)cccc2ccoc12 N1(C(C(C(=O)OC)C)=O)CCOC2CN(C(=O)Cc3cc(F)ccc3Cl)CC12 C1(CC(=O)NC2C(CC)C2)CCCCN(C(=O)CCc2ccncn2)C1 C1(F)(C(N2C(C(=O)NCC(CO)OC)C=CC2)=O)CC=CCC1 C1(CCNC(c2cc(C(N)=O)[nH]c2)=O)CCCCN1C(=O)COCC(F)F Cc1cc(N)cnc1C(N1CCC2CC12C(=O)NCCc1ccon1)=O N=c1[nH]cncc1C(=O)NCc1ccsc1C(=O)NCC1CC(CO)CO1 CC1CCN(C(C2(c3cc[nH]n3)CCC2)=O)CCN1C(=O)CCC1CCCN1C N1(C(CC2OCCN(C(C)=O)C2)=O)C(C)CN(C(c2sccc2F)=O)CC1C Cc1ccc2[nH]cc(CC(=O)N(C3CN(C(C4CCC(C)NC4=O)=O)C3)C)c2c1 N1(C(C2(C#N)CC=CC2)=O)CCCCC(CCC(=O)NC2(CO)CC(F)(F)C2)C1 N1(C(c2c(=N)[nH]cnc2)=O)CCC2C(CCCN2C(=O)Cc2ccc(O)nc2)C1 C1(C)(CNC(c2ccn(CCNC(C(C)SC)=O)c2)=O)CSC(C)=N1 CC1CC(CNC(C2(NC(c3nccnc3N)=O)CC(F)(F)C2)=O)CCO1 c1(C(N2CCCCC(CNC(c3cc(C)[nH]n3)=O)C2)=O)cc2ccoc2cc1F N(C)(C(=NCCc1ccc(F)cc1)NC1CCCOC1)Cc1scc(C)n1 C1CN2CCCCC2CO1.N(C1=NCC2CCC(N1)C2)c1ncn(C)n1.C(N)=O C1(C)(C(N2CC(CNC(CCc3nc(C)c(C)o3)=O)C(C)C2)=O)CCC(O)CC1 N(C(=NCCSC)NCCN1CCC(C)CC1)CCN(C(C)=O)CC c1(C(N2CC(C(=O)NCCC3CCCCC3C)(CC)C2)=O)cc2ccccc2[nH]1 CCCCCC(C)CC(=O)NC1CCC(NC(C2(N3CCOCC3)CC2)=O)CC1 c1(CC(=O)NC2C(NC(C3CC(C)(C)C3)=O)C2)ccc(C(F)(F)F)nc1 N1(Cc2nc(CC)on2)CCC2C(CCCN2C(c2cc(C)n(C(C)C)n2)=O)C1 N1(C(c2cc(CCC)ncc2)=O)CC(NC(c2c[nH]nc2C)=O)C(N=[N+]=[N-])C1 C1(O)(CC(=O)NCC2C(SC)CCC2)CCN(C(=O)CCC(C)=O)CC1 c1(C(=O)OCCc2ccc(Br)cc2)cc(Cl)cc(Cl)c1 c1(C(N2CC(NC(C3C(C)(C)C3)=O)C2)=O)ccc(CO)nc1.C(=O)(C1CC1)N N1(C(CC2=CCN(C)CC2)=O)CCC2(CCCN(C(=O)C=Cc3cc[nH]c3)C2)C1 N1(C(CSCC(=O)OC)=O)CCN(C(c2coc3c2CSC3)=O)CC(O)C1 C1(OC)CN2CCCC2(C(=O)NCC2CN(C(=O)CC(C)(C)OC)CCCO2)C1 c1(C(N2CCN(C(CCS(C)=O)=O)CC2C2CC2)=O)cccc2c1OCCCO2 C1(C(N(CCNC(c2cnc(C)o2)=O)CC2CC2)=O)CCC2(CC2)C1 N1(C(C(C2CCOC2)OCC)=O)CC2(CCCC2NC(C2(OC)CC2)=O)C1 c1(C(=O)NC2CC(N(C(c3c(OCC)nccc3)=O)C)C2)ccc(F)c(C)c1Cl c1(CN(CC(=O)NC(CCCNC(c2c(C)scc2)=O)C)C)cccc(Cl)c1 C(=O)(C(CO)c1ccccc1)OC(C)C(=O)NC1COC(=O)N1 C(=O)(N1CC(O)CCO1)c1c(CNC(c2n(C=C)nnc2)=O)n[nH]c1 c1(NC(c2c(CN=[N+]=[N-])cccc2)=O)cc(Br)c2[nH]c(=N)sc2c1 C1(CC(=O)C2CC2)CCCO1.CC1CC2(CC2)NCCC2(CC2)C(=O)N1 C1(C)(CC)CC(NC(c2ccc(C(N)=O)cc2)=O)CN1C(=O)CNc1nccs1 c1(C(N2CCC(C)C2C(=O)N(C)CC2CN(C)C2)=O)c[nH]c2cnccc12 N1(C(C(CCNC(CC(CC)C2CC2)=O)OC)=O)CCn2ccnc2C1C c1(C(=O)NC(CNC(=O)CSC)C2CC2)occc1C1CC1 N1(C(CCN(C(C)CS(C)(=O)=O)CC)=O)CC=CC1CN(C)C O=C(C1=NOCC1)NC1CCOCC1NC(c1ccccc1C1CCOC1)=O C1(CC)CN(C(=O)CC2CC2)CCN1C(=O)C(c1ccccc1F)C N1(C(C2CCN2C(c2c[nH]cc(Cl)c2=O)=O)=O)CCC2OCCC2C1 C1(CC)CN(C(c2cc(N)cc(O)c2)=O)CCN1C(c1nc(Cl)sc1C)=O c1(NC(c2n(C)ncc2S(C)(=O)=O)c2nnnn2CC)nccc2ccncc12 C1(CCCNC(C2CC2CF)=O)CCN(C(C2(C3CC3)CCCO2)=O)CC1 C1(NC(c2ccc(C(C)C)c(Cl)c2)=O)CC2CC1CN(C(=O)CNC(N)=O)C2 c1(C(N(CC(C)O)CCNC(C(CCOC)C)=O)=O)ccc2c(c1OC)CCC2 C#Cc1cnc(C(=O)NCC2CCCN(C(=O)Cc3ccoc3)CC2)c(C)c1 C(=O)(CC(=O)NCC1(O)CN(C(c2cc(C3CCC3)no2)=O)C1)OC Cc1cnc(NCC2(CO)CCOC2)c(S(=O)(=O)NC2CCCC(C)(C)C2)c1 C1(NC(C(N2CCC(O)CC2)C)=O)CCC(O)CN(C(=O)CCC(F)(F)F)C1 C(=O)(C(=O)CC(C)CC)N(C)CC1(O)CCCN(C(CC)=O)C1 C1(CCOC)CCN(C(C2CC(N(C)C(C3COCCO3)=O)C2)=O)C1 CCC(CC(=O)OC(c1c(F)ccc2c1OCO2)=O)CC(F)(F)F C(CCCC(F)(F)F)NC(C(c1cn(C)nn1)NC(c1n[nH]c(CC)c1C)=O)=O C1(NC(c2ccc(CO)o2)=O)COCC1NC(C1CCOC1)=O C(C)(C)(CC(N)=O)NC(C(C)N(C(C(C)NC(COC)=O)=O)C1CC1)=O C(=O)(C1CCCc2c(Br)cccc21)NCC1OCCN(CCCC)C1 n1(C(C)C)ncc(C(=O)NC2CC(CNC(=O)CC3CCC(=O)N3)C2)c1N CC1CC(NC(c2conc2C2CCC2)=O)CN1C(=O)CN(c1ncccn1)C c1(CC(=O)N(CCOC)CCNC(=O)C2CC2)ccnc(Br)c1 c1(C(=O)NCC2(O)CN(C(C3CN4CCN3CC4)=O)C2)ccc2c(c1O)CCC2 C1(C(N2CCC(N(C(=O)C(C)=CC3CC3)CC)C2)=O)CC12CCCC2 c1(C(=O)NC(CC)CN(C(=O)CCCC2CCC2)C)nccc(C)c1N N1(C(c2cnc(CCC)s2)=O)CCC2CCC(C1)N2C(=O)C(O)Cn1cncn1 CCCCCCCCCC(CC)C(=O)NC1CCCC1CNC(C1(CC)CC1)=O N1(C(CC)C)C(=O)NC(c2cc(OC)cnc2F)C2=C1CC(C)CNC2=O C(N=c1cc(NCCS(=O)(=O)N(C)C)nc(C(C)C)[nH]1)c1cc(CC)no1 N1(C(C2CN(C(C)=O)C2)=O)CC(NC(=O)Cc2n[nH]cc2Br)CC1(C)C Cn1nc(Br)c2c(N3CCCC(c4ccc(Cl)s4)C3)ncnc12 c1(CCC(=O)NCCN(CCC(C)C)C(C2CCN(C(N)=O)C2)=O)cccnc1Cl N1(C(C(C)(C)CC2CC2)=O)CCC2CCCN(C(=O)Cn3nccn3)C2C1 Cc1[nH]ccc(=NC(=O)Nc2cc(C(=O)O)c3cccnn23)c1Cl C1(C(=O)N)CC2CCC1C2.Cc1cnn(CCC=CCNC(C2(CCl)CCC2)=O)c1 CCC(=O)CCC(=O)NC1CC(C(F)C(=O)NCC2(C#N)CCC2)C1 c1(C(=O)NCC2COCCN(C(c3c(C)snc3)=O)C2)ccc2c(c1)COCC2 c1(C(=O)OC)ccc(CCNC2CC(OC)C2)cc1 CC1=C(C(=O)NCC(CNC(c2cnnc(O)c2)=O)C(F)(F)F)CCC1 c1(CNC(c2sccc2NCc2cccc(I)c2F)=O)ccc(F)cc1O C1(C(=O)NC2C(C)CCN(C(c3cc(OC)ns3)=O)C2)(OC)CCC(F)(F)CC1 c1(C(=O)NCC(CC)NC(=O)C(C)N(CC(F)(F)F)C)ccc(=N)[nH]n1 c1(OC)ccc(Cl)c(Cl)c1C(N1CC2(NC(=O)Cc3ccco3)CCC1CC2)=O c1(NC(=O)Nc2nccc(CC)c2)c(C#N)cnn1CC1CCCC1CCOC C1(C(=O)NC(C2CCCO2)CC)CCN(C(C2CC3(CC(OC)C3)C2)=O)C1(C)C C1(OC)CC(CNC(=O)C(C)c2ccsn2)N(C(=O)COCCF)C1 c1(SCC)ccc(CC(=O)N(C2CCN(C(c3ccccn3)=O)C2)C)cc1 CC(C)CC(C)(CNC(=O)CCc1cccc(O)n1)NC(=O)C(C#N)C1CC1 Cc1ccc(C(F)Cl)cc1C.c12ccc(C)c(c1)CC(=O)OC2 CCC(C(=O)NC1CC(NC(=O)Cn2cncn2)C1)c1ccccc1 C1(NC(=O)C=Cc2ccncc2)CC2(CCCCN2C(C2CCCCC2)=O)C1 C12(C(=O)NCCC(=O)OC(C)C)CCN(C(c3cc(CO)ncn3)=O)CCC1C2 CCCCCCCCC(=O)N1CCNCC1C=Cc1ccccc1 c1(CC(C)N(C)Cc2ccc(C(=O)OCC)o2)ccc(Br)cc1 c1(N(CCC(=O)OC)C(=O)CCNC(c2cccnc2)=O)ccccc1 C(CNC(=O)CCc1cc(Cl)cs1)(CC(F)(F)F)NC(C(C)c1ccco1)=O C(=O)(CCC(C)SC)N(CCC(=O)NC(c1ccccc1)CC)CCO c1(OCC)ccccc1CC(=O)OCC1CCN1C(=O)C=CC=CCCCCC c1(CNC(=O)NCc2ccc(OCCCOC)cc2)nc(NCC#N)cc(O)n1 CCC(CCCC(=O)N1CCC(N2CC(O)C2)C1)NC(c1n[nH]c2ccccc12)=O Cc1c(-n2cc(NCCC(Cl)Cl)cn2)cccc1[N+](=O)[O-] N1(C(CCCSC)=O)CC2C(CNC(c3ccc(N(C)C)cc3)=O)C2C1 CC(=O)C(C)CC(C)C(=O)N1CC(N(C)C(C2C3COCC23)=O)C2(CC2)C1 C1(ONC(CN(C(=O)CCCNC(C)=O)CC)=O)CCC(O)CC1 C12(C(=O)NC(C3CCOCC3)C#C)CC(CN(C(C3CCC(O)CN3C)=O)C1)C2 c1(C(=O)NC2CCCCN(C(c3cc(F)cc(Br)c3)=O)C2)c(F)cc(Cl)cc1Cl c1(NC(C2(CNC(C=CC=CC)=O)CC2)=O)cnc(F)c(C)c1 c1(C(N2CCC(CN(C(C(CC)C(C)O)=O)CC)CC2)=O)c(C)cc(C)oc1=O CN1CCC(C2CCN(C(C3CCOC(C)(C)C3)C(=O)NC(C)(C)C)C2)CC1 CC(C)C(C(=O)NC1CCC12CN(C(=O)CN(C)C)C2)S(=O)(=O)C1CCCCC1 C(C)(CC(C)NC(=O)CN(C(=O)C(C)C)C)NC(C(C)=C(CC)C)=O C1(NC(C(C)=O)=O)CCCC2CN(C(c3cc4cccc(C)c4[nH]3)=O)CC12 c1(N2CCC(N(CC)CC)CC2)nc(NCCC=CBr)c2ccsc2n1 N12CCC(C)(CC1)C(=O)NC1CC1CN(CC)CC2=O.C1(N(C)C)CCSC1 Cc1ccc(CN(C2CCCN(C(=O)CCC(C)C)C2)C)nc1 c1(C(=O)OC)n[nH]c(=NC2CN(C(=O)CCNC(C3CCCO3)=O)CC2(C)C)s1 C1(CC(=O)NC2CCCC(CNC(c3scc(C)c3)=O)C2)CC(=O)NC(=O)C1 N1(C(C2C(O)CCN(CC)C2)=O)Cc2ccccc2C(O)C1.C1(=O)CS(=O)(=O)N1 c1(OCCC)ccc(S(=O)(=O)NC2C3CN(C(=O)C(O)C(C)C)CC23)cc1 C#CC(C)(C)C(=O)NCc1ocnc1C(=O)NC1CCCC(c2ccccc2)C1 c1(C(N(C2CCC(NC(c3cc(C)c(C)[nH]3)=O)CC2)C)=O)cccc(F)c1F c1(OC)cc(NCCCCN2CCNCC2)c(OC)cc1Cl n1(CC)nc(C)c(C(=O)N(CCNC(C2CCCCS2)=O)C(C)C)c1Cl c1(C(=O)NC2(C)CN(C(C3CCOC3C(F)F)=O)C2)n[nH]c2cc(Cl)ccc12 N1(C(c2c(CCC)[nH]cc2)=O)CC(NC(c2cc(Cl)ns2)=O)C(SC)C1 Cc1cc(Br)ccc1CC(=O)Nc1cccnc1C(=O)N(C)C c1(CCO)ccc(CO)cc1.CC(CCCS)(CO)c1ccccc1 N1(C(Cc2nc(C)oc2)=O)CCN(C(c2cnc(C)n2C(F)F)=O)CCC1C c1(C2C(NC(C3CC(NC(CCOCCOC)=O)C3)=O)C2)nc2ccccc2[nH]1 N1(C(c2cnc(OCC)nc2)=O)CC2CCCC(C1)N2C(=O)C(C)CC(C)C N1(C(CSCCC)=O)CCC2(CCCC2NCc2cc(C)ns2)C1 N1(C(c2nccc(C)c2)=O)CC2CCC(C1)C2NC(c1cc(F)c[nH]1)=O O=C(CCC(F)(F)F)N1CCCC(C(N2CCN(C3CCC3)CC2)=O)CC1 C1(CNc2c(Br)cc(C)c(F)c2)Cc2ccc(C)cc2C1 c1(CC(N2C(CN)CCC2)=O)cc(Br)ccc1C.CCC1CNC1=O CC(C)S(=O)(=O)c1ccc(NC(c2cc(Br)c(O)cc2F)=O)cc1 C12(NC(CC(C)F)=O)CC3CCC(C1C2)N3C(=O)Cn1cc2ccccc2n1 CC1CCCCN1CC(=O)NC1CC(CC(=O)NCC(C2CCCO2)O)C1 C=CC(F)(F)C(=O)NCCC1CC(C(N2CC(OC(F)F)C2)=O)C1 N1(C(C2(C=C)CCC2)=O)CCN(C(=O)C(N2C(=O)CCC2=O)C)CC1 c1(OC)ccc(C(=O)NC2CC(C)(NC(C3CC(C(N)=O)C3)=O)C2)cn1 C1(C(N2CC(C(C)NC(c3ncn(CC)n3)=O)OCC2)=O)CNC(=O)CC1(C)C N1(C(CC(C(C)OC)NC(C2(c3ccccc3)CC2)=O)=O)Cc2c[nH]nc2C(C)C1 c1(C(N2CCC(N(C(C3CC3C3CCCC3)=O)CCO)CC2)=O)ccc([N+](=O)[O-])o1 C1(C(=O)NCCCC(C)NC(C(CC)SC)=O)CCC(=O)N(C)C1 N1(C(C(CCC)NC(C)=O)=O)CCC2CN(C(c3cc(F)cnc3Cl)=O)CC12 C(C)(CC(=O)NCCOCCOC)NC(CSCC#C)=O c1(C(N(CC(=O)N(CCOC)CCN)C)=O)ncc(C)cc1F.C(C)(=O)N Cc1oc([N+](=O)[O-])cc1C(N1CCC(C)C(NC(=O)CCS(N)(=O)=O)C1C)=O N1(C(CC=CC)=O)CCCC(C)(CNC(=O)C(C(C)O)NC(=O)OC(C)(C)C)C1 C(C1CCCC1)=C(C)C(=O)NC1CC(N(C(=O)CCNC(=O)OC(C)(C)C)C)C1 c1(C(=O)NC(C2(O)CN(C(C3CCC(C)C(C)C3)=O)C2)C)ncc(C#N)cc1Cl C1(N=c2nc[nH]s2)(CNC(C2CCc3nnc(O)n3C2)=O)CCCCCC1 C1(C(=O)NCC2(F)CC(CNC(c3n(CC)ncn3)=O)C2)CCn2nnnc2C1 CC(C)C(C(C)NC(=O)CCn1cnnn1)NC(c1conc1C1CCC1)=O c12cccnc1C(=O)N2.C1(N(S(C)(=O)=O)C2CC2)COC(C)(C)C1 C(=O)(CCCC(C)=O)NCC(CC=C)NC(c1cnc(C)n1C)=O C(=O)(C(C(C)(C)C)N(C)C)NCC(CCOC)NC(c1cnn(CCO)c1C)=O C(=O)(C1=Cc2ccccc2OC1)NCC(C)NC(=O)C(C)C(C)c1ccc(F)cc1 C(CCN(C)C)(C(=O)NC(c1ncc[nH]1)C)NC(CC1CCC(C)O1)=O c1(CNC(=O)C(N2CCCC23CC3)C2CC23CCC3)cc(Cl)cc(Cl)c1 C(CCCCC(=O)N1CCC1C1CCOCC1)NC(c1ncn(C(C)C)n1)=O Cc1nc(CC2CC2)sc1C(=O)NC12CC1CN(C(C1CC1F)=O)C2 N1(C(C2CCC(NC(C(C)(C)n3cncn3)=O)C2)=O)CC2CCC2(C)C1 CC1(C)C2CN(C(c3cc4cccnc4[nH]3)=O)C(CN3CCC(F)(CO)CC3)C12 c1(C(=O)NCCC2CCCN(C(CCc3cnn(C)n3)=O)C2)cccc(Cl)c1N C1(CCNC(c2c(C)ncs2)=O)CN(C(=O)CC2CC=CCC2)CC1C c1(CC)cscc1C(=O)NCCC(=O)NCC(C)C(=O)OC N1(C(CC2CCN(C(C)C)CC2)=O)CC(N=c2ccnc(N3CCOCC3)[nH]2)C1 C(C#Cc1cccc(Cl)c1)NCC1CCC(NC(CCCc2n(C)cnn2)=O)C1 c1(-n2cc(C(CC)NC(C3(Cl)CC3)=O)nn2)cccc(CO)c1 Cc1cc(C)c(CN=c2[nH]c(CC(c3ccccc3)O)ns2)c(C)c1 c1(C(=O)NCCCCCC(=O)OCC)cc(N)c(F)c(F)c1Cl C1(CC(=O)N(CCCNC(C2(CC)CCC2)=O)CCO)SC(=N)NC1=O c1(C(=O)NCC(CNC(=O)Cn2cnnc2O)OC)cccc(N)c1O N1(C(C2C(OC)CCC2)=O)CCC(O)(C(C)NC(=O)CN2CCC(F)(F)C2)C1 CC(C)CC(C)CC(=O)N1CCC(C(C)NC(c2csc(CO)n2)=O)CC1 N1(C(C(C)SC(C)C)=O)CC2CCCN(C(C3CC4COCC(C3)C4=O)=O)C2C1 C12(C(N3CCC(c4cn(C(C5CCCOC5)C)nn4)C3)=O)CCCCC(F)(C1)C2 C1(C(=O)NC(c2ccc(C)nc2)C)C2CC3C(C2NC(c2cnc(O)o2)=O)C13 c1(C(=O)NCc2cn(CCNC(C(CCC)N(C)C)=O)nn2)ccc(C)cc1F CN1CCN(C(C2CCCCO2)=O)C(CNC(C2CC3CCC2C3)=O)C1 c1(C(N2CCN(C(CC3(NC(C)=O)CC3)=O)CC2)=O)cnc(Cl)c(Cl)c1 c1(CC(N2CC(C)C(NC(c3cccc(=O)n3C)=O)C2)=O)cc(F)cc(F)c1 C12(NC(c3c(=N)c(Br)c[nH]c3)=O)CCCC1CN(C(C1C3CCCC13)=O)C2 c1(OCCOC)ccc(C(=O)NC2CN(C(c3nccn3C)=O)C3CC23)cc1 CCCCCC(O)CC(=O)N(CCCNC(C1CCN(C)C(=O)C1)=O)CCO C1(C(N(CCC(=O)NC)CC)=O)CCN(C(=O)C(C#N)C(C)(C)C)C12CCC2 Cc1noc(C)c1CN1CCC(NC(c2cc(Br)c[nH]2)=O)C1 CC1CCCN(C(c2cccc(N)n2)=O)C1CNC(=O)C(C)(C)c1sccc1Cl C(=O)(C1=CCCCO1)NCCCC(C)(C)NC(c1cc2c(s1)CCC2)=O CS(=O)(=O)c1cccnc1CN1CCC(c2ccc(Br)nc2)CC1 c1(C(N2CC(NC(CC(CC)(C)C)=O)C(C)CC2)=O)sc2ncccc2c1N C1(NC(c2c(OC)cc(F)c(F)c2)=O)CS(=O)(=O)C12CCCC2 Cc1cc(C(=O)NC(C(=O)N(C)Cc2nncs2)C(C)C)cc(C)c1 CCCCC(CC)CC(CNC(=O)C(F)n1cccn1)CC C(=O)(CCCC(CC)NC(=O)CCc1cc(C)on1)N(CCCC=C)C c1(CNC(COC)=O)n[nH]c2c1CN(C(=O)Cc1cn3c(C)csc3n1)CC2 C(=O)(C(C(C)(C)C)N(S(C)(=O)=O)C1CC1)N(CCCCN(C(C1(C#C)CC1)=O)C)C c1(C(=O)NC2CCC(F)(CNC(C(CC)C)=O)C2)cc(F)cc2ccccc12 c1(-n2ccc(CNC(C(=O)NCC3(CCF)CC3)=O)n2)ccc(C(F)(F)F)cc1 C1(C(=O)NCc2cnn[nH]2)(OCC)CCN(C(=O)CC(C)C)C1 N1(C(C(N2CCN(C)CC2)C)=O)CC=CC(NC(c2csc(CC(F)F)n2)=O)C1 c1(SC)cc(N2CCN(C(c3ccccc3C#N)=O)CC2C)nc(SC)n1 c1(C(N2CC3(C(NC(c4n(C=C)nnc4)=O)CC3)C2)=O)c([N+](=O)[O-])c(C)nn1C C1(C(N(C(CC)CC)C)=O)(CC)CCN(C(c2cccc(OC)c2O)=O)CC1 C1(C(N2CCC(NC(c3c(CCC)n(CC)nn3)=O)C2)=O)OCC2CCCC12 c1(C(N2CCCC(N(C(C(C)=C3CC3)=O)C)C2)=O)cc(C)c(F)cc1Br c1(CNC(CC(=O)NC2CC(F)(F)C2)Cc2cccc(Br)c2)c(Br)cncc1Br c1(C(COC(c2c(CC)n(C)nc2)=O)=O)ccc(Cl)c(Cl)c1 Cc1ccc(Cl)c(C(=O)NC2COCC2NC(C2COCCO2)=O)c1 c1(C(C(=O)N(C2C3CN(C(=O)CCC4CC4)CC23)C)O)cc(F)c(F)cc1F CC(CCC(C)(C)C)C(=O)N(C)CC1CCCN1C(c1csnn1)=O N1(C(C(CSC)OC)=O)CC(F)(F)CC1CNC(=O)CC1CCC(O)C1 C(CC(=O)NCC1CCC2(CC2)C1)(C(C)OC)NC(c1cncc(OC)c1)=O c1(N2CCCC(C)C2)ccc(Cl)cc1NC(=O)C(N1CCC(F)C(O)C1)=O c1(OC)cc(C(N2CCN(CCNC(=O)C=C3CCCCC3)CC2)=O)ccc1O O=S(=O)(c1ccns1)N1CCN(Cc2ccc(OCl)cc2)CC1 C1(CNC(C2(C(C)C)CCC2)=O)CC2CC1CN2C(C1CCO1)=O CCC(C(=O)NC1CC(F)CN(C(=O)C(=O)NCC(F)F)C1)C(C)(C)CC c1nccc2cc(Br)ccc12.Cc1noc(C(C)(C)CNC(=O)C(=O)N)n1 CCC(C(=O)NCCn1cc(C(N2CC(CC)(CO)C2)=O)nn1)C(C)C n1(C(C)C)cc(CNC(C2CCN2C(=O)C=CCF)=O)cn1 Cc1ccc(C(F)F)c(C(=O)NCC(n2cc(-c3ccn(C)n3)nn2)C)c1 N12CCCC(CC1)n1cc(nn1)C2(C)C.CC1(C)CC1NCCS(C)(=O)=O C1(CC(=O)NC2(CCNC(Cc3c(C)nc[nH]3)=O)CCC2)CCC(=O)NC1 c1(C(=O)NCC2(C)C(NC(c3n(CC)ncn3)=O)CCC2)cc(Cl)cc(Cl)c1 C(CC(=O)NCC(C1CCOC1)NC(=O)CN(C)C(C)C)NC(C)=O c1(C(=O)NC2(C)CN(C(CCN(S(C)(=O)=O)C)=O)C2)nccc2cc[nH]c12 C=C1CCN(C(c2cncnc2C)=O)C(C(=O)N(C(COC)CC)C)C1 CC1C(C)N(C(C2CC(C)(C)C2)=O)CCN1C(c1nn2c(c1Br)CCC2)=O c1(N2CCN(C)C(CNC(c3ccnc(F)c3)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 c1(C(=O)NC2CCCN(C(Cc3cc(CC)nn3C)=O)C2)c(O)cccc1O C1(NC(c2ccc(C(F)(F)F)cn2)=O)CC12CC(NC(C1(F)CC1)=O)C2 CC(C(=O)N1CC(N2CCCC2=O)C1)(C1CCC1)NC(C1(c2ccno2)CC1)=O C1(C(=O)NCC2CCCN(C(CCOC(C)(C)C)=O)CC2)CC2CSCC(C1)C2 c1(C(N2CC(C(N(C(C)C3CC3)C3CC3)=O)C(C)CC2)=O)cc2cccnn2c1 CC(C)CC(F)C(=O)N(CC(C)(C)NC(=O)C(C(C)C)n1ccc(C2CC2)n1)C c1(C(=O)NCC2(C)CCN(C(CC(=O)OCC)=O)C2)ccc(N(C)C)cc1F C#CCCCCCCN=C(NCC(F)(F)CO)NCC1CC1(c1ccccc1)C C1(CC(=O)NCC(C)(C)N(C)C(=O)OC(C)(C)C)CC2CC1CC2=O C(C)(CCCNC(=O)CCCNC(N)=O)NC(C(C1CCCC1)OC)=O CCC(C)CC(C(=O)NCC1(C2CC2)CCCO1)NC(=O)CN(C)C C(=O)(C1CCCc2nc[nH]c21)N1C(CNC(=O)CC2CSCCO2)CCC1 Cn1c(SNCc2nnn(C)n2)nc2ccncc12 c1(C(=O)NC(COC)CNC(C2(C)CCCO2)=O)c(C)ccc(C)c1N C1(C#N)(C(=O)NCC2(NC(c3nc(C(C)C)oc3)=O)CCC2)CC12CCOCC2 c1(C(=O)NC2C(CNC(c3c(C)oc(Br)c3)=O)C2)ncnc(O)c1F N1(C(CCCOCCC)=O)CC2CCN(C(=O)C(N3CCC(O)CC3)C)C2C1 C1(C(=O)NC(C)CCNC(c2cnc(C(C)(C)C)o2)=O)CCC(C2CCC2)CC1 C1(N2CC(C)OCCC2)CC2(C1)CN(C(c1ccc(N(C)C)nc1)=O)C2 CC1(C)C(CNC(=O)CC2CCCC2(F)F)CCN1C(C1CCCNS1(=O)=O)=O CC1CCN(C(=O)C(=O)NC2(C)CCN(C(=O)Cc3nc(Cl)cs3)C2)CC1 C1(C(=O)NC2CN(Cc3nc(CCOC)on3)CC2(C)C)CCc2nccn2C1 C1(NC(=O)COc2ccccc2)CC2CC(NC(C3CCC(F)(F)C3O)=O)C1C2 CC1CN(C(c2ccc(F)s2)=O)CCC1CNC(C1(C(C)(C)C)CCC1)=O C(CCC(=O)NCCC1CCC(C)C1)NC(=O)NC c1(SC)cc(C(=O)NCCCCCCn2cc(C3COCC3O)nn2)c(C)o1 C(=O)(NNc1ccc2c3c(cccc13)CC2)C1(N)CCCC1 C(CC(=O)NCC(CC1CC1)CO)(C1CC1)NC(C=CC=CCC)=O Cc1[nH]ccc1C(=O)NC1CCC1NC(c1nocc1Br)=O c1(C(N2C(C(C)NC(C(C=CCCC)O)=O)CCC2)=O)nc2ccccn2c1F C1(C(N2CC(C#CC)C2)=O)CCC2(CC2)N1C(C1CC2(CCC2O)C1)=O c1(C(C(C)C)OC(=O)CC2COCC(C)(C)O2)nc2ccccc2[nH]1 CCC(C)(CCNC(=O)C=CSC)NC(c1cc(C)nn1C)=O N1(C(COCCNC(C2CCSC2)=O)=O)CC=CC(O)C1 c1(Cn2cc(C(CSCC)C)nn2)ccc(C(N2CC(C(=O)O)(OC)C2)=O)cc1 N1(CC(=O)N(C(C)C)C2CC2)CC2CC1CN2C(c1cnn2c1CCC2)=O C1(CC)(CNC(C2CCCC(CC)CC2)=O)CCCC(=O)N1 C1(C(=O)NC2(C#C)CC2)CCCCN(C(c2cccc(C)c2C)=O)C1 c1(C(=O)NC(C2(O)CCN(C(C3(O)CCSC3)=O)C2)C)csc2c1CCCC2 N1(C(C(CC)(C#N)CC)=O)CC(NC(=O)C(F)OC(F)(F)F)CC12CCCC2 N1(C(C2=C(C)CCC2)=O)Cc2[nH]nc(C(=O)NCC3OC(=O)CC3(C)C)c2C1 [N-]=[N+]=NC1CN(C(C2CN3CCN2CC3)=O)CC1NC(C1(N2CCCC2)CC1)=O c1(CC(CO)NCc2cc(COC)on2)ccccc1F N1(C(CCC=C(C)C)=O)CC2CCC(NC(C3OC(C)CC3C)=O)CC2C1 C(=O)(CCCCCF)N1CC(n2cc(C(CC3COCC(C)O3)O)nn2)C1 c1(CC)cncc(C(N2CCCC2(C)CNC(=O)CCc2ccn(C)n2)=O)c1 C1(N(C(=O)CC#N)C)CN(C(=O)Cc2c(F)cccc2F)CCC1O CS(=O)(=O)c1ccnc(NC2CN(C(=O)C=CI)CCC2C(F)(F)F)n1 CC1CN(C(=O)C(=O)C(C)(C)C)CCC1C(=O)NCc1occc1C(N)=O n1(CC(=O)N(CC(O)CNC(C23CCCC2C3)=O)C)cnc2sccc2c1=O CN1C2CCC1CN(C(=O)CC=CCNC(=O)C1=C(Cl)CCC1)C2 CC(C)(C)C(=O)CCC(=O)N1CCOCC1c1nc[nH]n1 CN1CCC2CN(C(C3CC(F)(F)CN3Cc3ccnc(Cl)c3Cl)=O)CC2C1 C1(CCC)CN(C(c2ccc(C(F)F)cc2Cl)=O)CCN1C(C1CC12CC2)=O c1(NC(C2N(C(c3cc(C)c(Cl)nc3)=O)CCCC2)=O)cc(F)cc(C#N)c1 Cc1oc2ncnc(O)c2c1C(=O)NCC(C)(CO)NC(c1ccncc1)=O c1(C(=O)NC2C(C)CN(C(c3c(Cl)csc3Cl)=O)C2)cc(C2CC2)cc(F)c1 c1(C(N(CCN(C(C2C(C(=O)NCC#C)C2)=O)C)C(C)C)=O)cnccn1 Cc1cc(C)c(C(N2CCCN(C(c3cnc(S)[nH]3)=O)CC2C(C)C)=O)cc1C c1(C(=O)NC2CCC(N(C(=O)CCc3nccs3)C)C2)cc(Cl)ccc1O N1(C(Cc2c(OC)nccc2)=O)CCC2CN(C(=O)CCc3ncc[nH]3)CC2C1 C1(C(=O)NCC2(NC(CSCCC)=O)CCC2)CSCC(=O)N1 C1(c2ccccc2)(CNC(N2C(CC(=O)OC)CCC2)=O)COCCO1 N1(C(c2nc(C)oc2)=O)CC(NC(C2CCC(=O)NC2)=O)C2(COC2)C1 Cc1ccc2n[nH]cc2c1NC1CCN(C(=O)OC(C)(C)C)C1C(C)(C)C Cc1c(C(=O)NC(C)CNC(=O)Cc2ccc(Cl)cc2Cl)[nH]c2c1CCCC2 CC(CC(=O)NCC1(C)CCN(C(=O)Cc2c(O)ncnc2O)C1)CC(F)(F)F c1(CC)cc(C(N2CCC(CNC(=O)CC3(O)CCCN(C)C3)C2)=O)ccc1O c1(OC)cnc(C(=O)NC(C)CC2CN(C(=O)C(C)(C)C3CC3)C2)c(OC)n1 CC(CC(=O)N1CC(C)(C(N2CCC(C#N)C2)=O)CC1(C)C)C(F)(F)F C(=O)(CC(C)C(F)(F)F)NC1CCN(C(C2(C=C)CCC2)=O)C1 C1(OC)CCCN(C(=O)NC2CCN(C(c3cc(Cl)ccc3C)=O)C2)C1OC c1(C(=O)NCC2C=CC(NC(CC#N)=O)C2)nnc(O)c2c1CCCC2 C1(NC(c2cn(CC)nc2)=O)CCC2CN(C(c3conc3C)=O)CCC2C1 Cc1ncc(Cl)cc1C(N1CCC(NCc2cnc(O)c(Cl)c2)C(F)C1)=O Nc1cccc(C(N2CCCOC(CCNC(=O)CC3CCSCC3)C2)=O)c1F N1(C(c2ccncc2F)=O)CCCC2(C1)CN(C(C1CCCOC1)=O)CCO2 CC1(C)CCCC(O)(C(=O)NCC(C2CC2)NC(=O)Cc2ccccc2Cl)CC1 c1(C(=O)NCC(CNC(c2c(C)n(CC(C)C)nc2)=O)CO)cc2occc2s1 c1(OC)ccc(CCC(=O)NCC2(F)CCN(C(=O)Cc3cnoc3)C2)cc1C C1(NC(=O)CC=C(Cl)Cl)COC2(C1)CN(C(c1ccc(O)cc1O)=O)C2 C1(C)CCCCC1CN.Cc1oncc1C(=O)NCC(C(=O)C(C)C)=O N1(C(CCNC(CC2CCC(=O)C2)=O)=O)CCC2(CCC2)C1 c1(CNC(=O)NCC2(O)CCOC2)cccc(C2CC2)c1F c1(C(=O)NC2(CNC(c3nn(CC)c(C4CC4)c3)=O)CC2)ccc(N(C)C)cc1 N1(C(c2ccc(CC)cc2)=O)CC2CCCC2(N=c2[nH]nc(CO)s2)C1 C12(NC(C3N=C(C)SC3)=O)CCC(C1)N(C(c1ccc(CNC(N)=O)cc1)=O)C2 C1(C(=O)NCC(C)NC(Cc2cc(OC)no2)=O)CCc2ccccc2CC1 N1(C(C=CCN(C)CC)=O)CC2(CCCC2NC(=O)CNC(c2ccsc2)=O)C1 Cc1nc(C(N2CC(C)(C(=O)NC3COCC3O)C2)=O)sc1C N1(C(c2c(C)cc(Br)cn2)=O)CCC2(CCC2NC(C2C3CC4C(C3)C24)=O)CC1 N1(C(C=CCC)=O)C2CCC1CC(CNC(C1(c3ccnc(Cl)c3)CC1)=O)C2 CC1CN(C(=O)CSCC(F)F)CC(C)CN1C(C1CCNC1=O)=O c12ccc(cc1Cl)C(=O)NCC1(CC1)CCNC(=O)C=CC2.c1(CC)cnoc1 c1(C(N(CCNC(c2cc(OC)ccn2)=O)CC)=O)cnc(SC)nc1Cl c1(C(C)C)cc(C(=O)NCC(O)CNC(C2(CCF)CCC2)=O)no1 c1(N2CCN(C(c3c(F)ccc(O)c3F)=O)C3C2C3)ncnc2c(Br)cccc12 C(=O)(C(C)(C)CCSC)NCC1(CCNC(C2CCN(C(CC)=O)C2)=O)CC1 c1(C(N(C)CC2C3CN(C(CCCC)=O)CC32)=O)cccn(C2CCC2)c1=O C1(NC(c2ccn(C3CC3)n2)=O)CC2CCC(C1)N2C(c1c(O)cncc1F)=O Cc1cc(Cl)c(C(=O)NCC2CCN(C(=O)CCCC3CC3)C2)cc1Br C(=O)(C(F)C(=O)NCC1CN(C(=O)C(C)OCCC(C)C)CCO1)OCC c1(ONC(CNC(CN(C2CC(O)C2)C)=O)=O)cccc(Cl)c1 c1(C(N(CCN(C(=O)CC2CCC(OC)CC2)CC)CC)=O)cc(Cl)cc(Cl)c1F c1(C(N)=O)cc(Br)ncc1NC(C12CC1CN(C(c1nc(Br)cs1)=O)C2)=O c1(C(=O)NC2C(NC(C3(C)CC=CCC3)=O)CC2)cc(F)cc2cnccc12 C=C1CCN(C(c2c(CO)n[nH]c2C)=O)C(C(N2CCCC2CCOCC)=O)C1 C1(O)(CNC(c2ccc(OC)cc2)=O)CCCN(C(=O)CSS(C)(=O)=O)CC1 c1(C(=O)OC)cc(C)c(NC(=O)NC2CCC(C)(C)O2)c(Cl)c1 c1(OC)ccc2nc(N3CCCC3C(=O)NC3CC(N4CCCC4=O)C3)sc2c1 CCC(C(=O)NC(COC)CO)NC(c1cncnc1)=O N1(C(CC2CC(C)C2)=O)CCN(CCCNC(=O)Cn2cnc(C#N)n2)CC1 C(CN=c1ccc(Br)c(S(=O)(=O)NCCC2CC3CCC(C2)C3)[nH]1)SCC c1(CC)c(C(=O)NCCCCNCCCNC(=O)CC2CCC3CC23)csc1C N1(C(c2ccc(NC)cn2)=O)CCC(NC(=O)COc2ccccc2)C12CCC2 c1(OC)ccncc1C(=O)NC1CCCC1C(=O)NC1CCCC12CC2 Cc1ccc(P(C)(C)=O)c(NC(=O)C(N2CCOC(C#N)C2)=O)c1 C1(COC)CN(C(C2(C#N)CC(=O)C2)=O)CCN1C(=O)Cn1nccc1C c1(C(=O)NCC(CNC(C(CC2CCCC2)OC)=O)O)cccc(Cl)c1[N+](=O)[O-] c1(Cn2cc(-c3c(COC)con3)nn2)cc(F)cc(S(N)(=O)=O)c1 N1(C(c2cc3nc(C)[nH]c3nc2)=O)CC(NC(=O)C=CCO)CC12CCCOC2 C(=O)(C1=CCCN(C(c2ccc(O)nc2)=O)C1)Nc1ncc(C)cc1Br C=CCC(CNC(=O)C=CCOCCOC)NC(c1occc1F)=O c1(C(=O)NC(C)CCNC(c2cc(F)c[nH]2)=O)cc(Br)nn1C c1(C(N(C(CNC(c2c(CC)nns2)=O)C)C)=O)cncc(F)c1Cl c1(CC)c[nH]nc1C(=O)NC1(CCNC(=O)C(C)Cc2cnn(C)c2)CC1 CC1CC(C(=O)NC(C)(C)C=CC(=O)NC2C(O)CC2O)CO1 C1(C(N(CCNC(c2cc(C)sn2)=O)C)=O)CCC2(CCCC2)C1 c1(OC)cc(C)ccc1C(N1CC(CC(C)NC(c2csc(C)c2C)=O)C1)=O c1(C(N2CC(C)C(NC(c3cncn(C)c3=O)=O)C2)=O)ccc(F)c2ccsc12 c1(NC(=O)NC2CCC(C(=O)NCc3n(CC)ncc3)OC2)cc2ccsc2n1C c1(OC)ccc(CCC(N2CCOCC2C(=O)Nc2nc(C)c(Cl)s2)=O)cc1Cl c1(CC2N(C(c3c(C(=O)OC)nns3)=O)CCOC2)ccc(Cl)c(Cl)c1 N1(C(C2CC(C(=O)OC)C2)=O)CCCC1C1CCN(C(=O)C=CBr)C1 Cc1nc(C(N2CCSCC2CCNC(=O)CCC(C)(C)C)=O)ccc1C#N C1(CNC(C(C)Cn2ccnc2)=O)CC2CCC(C1)N2C(c1cscc1F)=O c1(OC)ccc(C(c2nnnn2C2CC(F)(F)C2)NCCOCCO)cc1 CC(C(C)(C)C(=O)NCC=C1CCSCC1)NC(=O)CC1CSCCO1 O=[N+]([O-])c1ccc2[nH]cc(CC(C3CC3)NC3(C4CC4)CC3)c2c1 Cc1cc(N)c(C(N2CCCOC(CNC(=O)C=CC3CCCO3)C2)=O)cc1C N1(C(c2ccnc(C(F)(F)F)c2F)C(=O)NCC=C)CCNCCC1(C)C N1(C(c2ccc(Cl)c(C)c2Cl)C(=O)NC(CC)C)CCC2(CCOC2=O)C1 c1(C(=O)NC(c2cnc(OC)s2)C)cnc(OC(C)C)c(Cl)c1 O=C(CC(O)C(Cl)(Cl)Cl)NCC1(F)CCN(C(c2cc3ccccn3c2)=O)C1 Cc1cc(C(=O)NCC(CO)NC(C2CC2CC(C)C)=O)c2occc2c1 CC(O)C(C(=O)N1CCCC(NC(=O)CC2CCCC2(F)F)C1)N(C)C c1(CC)ncsc1C(=O)NCC1(CC(=O)NCCO)CC1.C1(C)CC1 c1(C(=O)NCC2C(NC(c3c(CC)nco3)=O)C2)cc(Cl)cc(F)c1N C1(N(C)Cc2ccccc2F)CN(C(=O)Cc2cnn(C)c2)CC1(C)C C1(CNC(c2c(C)cccn2)=O)CN(C(=O)C(C)(C)OCCF)CCCO1 CC(C(=O)N1CCN(C(c2ccc(C3CC3)cc2)=O)C(CC2CC2)C1)C(F)(F)F C1(C(=O)Nc2cnc(C)c(Cl)c2)CC2(CCN(C(=O)CN3CCCC3)C2)C1 c1(C(C(=O)NCCOCCNC(C2C(C)CCCC2)=O)O)cc(F)c(F)c(F)c1 N1(C(C(CC(=C)C)NC(C)=O)=O)CCC2CN(C(C3CCCC3)=O)CC2C1 N1(C(CCC2CC(NC(=O)C(F)CC3CCOC3)C2)=O)CCC(C#N)C1 C12(C(CNC(N3CCCC3c3cncc(Br)c3)=O)O)CCC(CC1)C2 C1(C(N2CC3(C(NC(CCC#C)=O)CC3)C2)=O)CCC2(CC1)CC(OC)C2 C(C(=O)NC(C1CCN(C(c2cnc(S)[nH]2)=O)C1)(C)C)(C(C)C)NC(=O)OC CN1CCN(C(C2CC2C2CC2)=O)C(CNC(=O)CCn2cc(Br)cn2)C1 C1(C(N2CCC(O)(CC#N)C2)C(=O)Nc2ccccc2Cl)Cc2nccn2C1 c1(C(=O)NCC(CC)NC(=O)CC2CC(=O)NC2=O)ccc(F)c(C)c1C#N C1(CC=C)(NC(c2ccccn2)=O)CCCN(C(=O)CC2CC=CCN2C)C1 CC(CCCCN=c1nc(C(F)(F)F)cc[nH]1)NC(C1(C)CCCS1(=O)=O)=O N1(CC(=O)NC(C)C(CO)NC(=O)Cc2cnc(C3CC3)[nH]2)C(=O)CN(C)C1=O C1(NC(CC(=O)NC2CC2)=O)CC2CCC1N(C(=O)CC(O)c1ccccc1)C2 c1(OC)ccc(-c2cn(CC3CC3)nn2)s1.C1C(=O)CCS1 C1(C(=O)NCC2CCC(F)(CNC(c3cn(C)nc3O)=O)C2)CCCC(C)(C)C1 C(=O)(C(CC)(CC)OC)NCC(CCCC)NC(c1ccc(C(C)=O)s1)=O c1(C(=O)NC(C(=O)NCCOCCF)C2CC2)ccc(F)cn1 N1(C(CCC(=O)NCC)=O)CCC12CN(C(=O)CCCc1ccncc1)C2 CC1(F)CN(C(=O)CC2CCCCC(=O)N2)CCN(c2cc(F)ncn2)C1 C1(CNC(C2N(C)CCC2)=O)CC2(CCC2)CN1C(=O)CC(=O)NCC1CC1 CC1CCCC(C(=O)NCCn2cc(C(N3CCCC3C(N)=O)=O)cn2)C1 c1(CC)ccc(C(N2CC3CC3(C(=O)Nc3cccc(OC)n3)C2)=O)cc1Br N1(Cc2c(C)ccc(C)c2)CCCC12CCN(C)CC2.C1S(=O)(=O)NC12CC2 C1(C(=O)NC2CC(C#C)C2)CSCCN1C(c1cc(C)c(C)[nH]1)=O c1(C(=O)NC2CC(NC(CCC(=C)Br)=O)C2)cccc(CO)n1 CCC(CC(=O)N1CC(C(=O)NCCNC(C2(F)CCCC2)=O)C1)C(F)F N1(C(CN(CCC)C)=O)CC(OC)CC(NC(=O)C=C(C)c2cccnc2)C1 N(C(=NCCCF)NCCCS(C)(=N)=O)CC1(OCC)CCSC1 N1(C(C(CC)C2CC2)=O)CCC(C)(CNC(=O)C=CCN2CCOCC2)CC1 C1(CNC(c2cc(CCC(=O)OC)c[nH]2)C(=O)OC)COCCN1C c1(NC(CNCC(C(C)O)(C)C)=O)cn2c(Br)cccc2n1 N1(C(CC)=O)CC(C)C(NC(c2cc(CC)cc(C)c2)=O)C(C)C1 c1(C(N2CC(CC)C(NC(C3(N(C)C)CCC3)=O)CC2)=O)cnn2ccccc12 O=C(CCCCCO)NC1(CO)CCCN(CC(=O)Nc2ncccn2)C1 c1(CC(=O)NCC2CCN(C(C(CC)OC)=O)C2)ccc(-n2ccc(O)n2)cc1 N1(C(CCOC(CC(C)C)C)=O)CCCC(CNC(=O)CN2CCC2)C1 N1(CC)CC(COC(c2cc(-c3ccccc3)ccn2)=O)OC1=O C1(c2ccc(Br)cc2)(C(=O)OC)CCN(C(=O)C(C2CCCCC2)C)C1 C1(CNC(=O)CC(O)C2CCCC2)CCCN(C(=O)C=CC2CCCO2)CC1 c1(C(CC)NC(N2CCC(CCCO)C2)=O)ccc(O)cc1 C(C1CCCN1C(=O)C(C)OCOC)=CC(N1C(CCC#C)CCC1)=O c1(C(C)=O)cn(C)nc1C(=O)NC1C2CN(C(c3ccc(C(N)=O)nc3)=O)CC12 c1(CC)c(C(=O)NC2CN(C(=O)CC3CC4CC4C3)CC2F)nnn1CC c1(C(=O)NCC2(C(=O)NCC(COC)O)CC3(CC3)C2)cccc(O)c1C C1(C(=O)NC(C2(O)CCC2)C)(CC)CCN(C(=O)CNC(C)=O)CC1 N12CCC3(CC1)CC3C2.N1(C(c2cscn2)C)CCOCC1CO.C1(C)=CCC1 CCCC(C(=O)NCc1ccccc1CNC(C1CC1C(N)=O)=O)OCC CC(CC1CC1)C(=O)NCC1CC(O)(CNC(C2(CCF)CC2)=O)C1 C1(C)(C(N2C(CNC(CC3C(C)=NN(C)C3=O)=O)CC2)=O)CC2(C1)CC(F)(F)C2 CC1CN(C(N2CCC2C2CCOC2)=O)CCc2ccc(Cl)cc21 C(=O)(C1CNc2c(C(F)(F)F)cccc21)NCC(CCOC)O CN1C(=O)CSC1=C(Cl)C(=O)NCC1CCN(C(=O)Cn2cncn2)C1 C(=O)(CCCS(N)(=O)=O)NC1CN(C(c2cnc(SC)nc2O)=O)CC1C C12(CC(C)(C)C1)C(=O)N2.c12ocnc1C(=O)NC2.C1(CC)CC(O)C1SC Cc1cc(C)c2[nH]c(=NC3CCCCC3CNC(=O)CCCCC(N)=O)sc2c1 C1(CNC(C=C(COC)C)=O)CC(O)CN1C(=O)CCN(C)CCO C1(CC)CN(C(=O)CCc2cc(SC)oc2C)CCN1C(c1cccc(O)n1)=O c1(C(=O)NCC(C2CC2)NC(c2c[nH]c(Br)c2)=O)nnn2c1COCC2 C1(NC(CN(CCOC)C)=O)CCN(C(=O)Cc2ccc(F)c(OC)c2)C12CC2 C1(CC(=O)Nc2c(C)nsc2)CCCCN1Cc1ccc(COC)cc1 C1(NC(C(F)=CCC)=O)CCC2(CC1)CC2NC(C1CCN1C(C)(C)C)=O n1(CC)cc(CC(=O)NC(c2nnnn2-c2ccccc2)CC2(C)N=N2)cn1 C1(NC(c2ccc(OC)s2)=O)CC2CN(C(=O)CCOc3ccccc3)CC2C1 c12nc(c(C)cc1Br)NC2c1nnnn1CCCF.C(C(C)C)OCCOC N(C(=NCCC1(O)CCC1)NC(C1CC1)C1CC1)CC1(C)C(C)CCC1 c1(C(N2CC3C(CNC(c4ccn(COC)n4)=O)(C3)C2)=O)ccc2oncc2c1 c1(CC)cc(C)ccc1NC(c1coc(CNC(C2(SC)CCC2)=O)n1)=O CC1CCN(C(=O)CC(=O)OC(C)(C)C)C1C(N1CCC(c2cnn[nH]2)C1)=O CCC(C)(C(=O)NC1CC2CCC1CN2C(c1cccn1C1CC1)=O)C(N)=O N1(C(c2ccc(CN(C)C)cc2)=O)CCCN(C(c2cc(C(F)F)no2)=O)CC1 N1(C(c2ccc(Cl)c(Cl)n2)=O)CC2CCC2(C(N2CCCC(Br)C2)=O)C1 C1(NC2C(Cc3n(C(CC)(C)C)nnn3)CC2OCC)CC2C=CCC(C1)C2 c1(C(=O)NC2(CC=C)CN(C(=O)CCc3scnc3C)C2)ncc(Br)cn1 C1(NC(c2ccc(CCC)[nH]2)=O)CN(C(=O)C(=O)NCC(F)F)C2(CCOC2)C1 N1(C(COCCC=C)=O)CC(F)CC1C(N1CCC(CC)(CO)C1)=O CC1CC(c2ccccc2)(C(=O)NC2CCC(NC(=O)CCC3CCC3)C2)C1 C(=O)(C(C)N(OC)C(=O)C(C)N(C(c1ccc(F)cc1)=O)C1CC1)OC c1(-c2ccc(Nc3ccnc(C)n3)s2)ccc2c(c1)NC(=O)CO2 c1(C(C)C)ccccc1C(F)(F)C(=O)N(C)C(c1nc[nH]n1)C C1(CNC(C=C(CCC)C)=O)(COC)CCCN1C(c1cncc(C2CC2)c1)=O Cc1ccc2[nH]c(CNc3ccsc3C(N3CC(CO)CC(F)C3)=O)cc2c1 C1(F)(C(N(CCN(C(C)C)C(C2NC(=O)NC2=O)=O)C)=O)CCN(C)CC1 c1(C(CC(=O)N(CCNC(C2(O)COC2)=O)CC)C)ccccc1C C1(C)(COC)CCN(C(=O)NC2(CC(=O)OC(C)(C)C)CCCC2)C1 Cn1ccc(C(=O)NC2CC(F)(CNC(=O)CNC=O)C2)cncccc1=O n1(CC)ncc2cc(NC(=O)NCC3CC(COC)C3)cnc12 C1(NC(c2[nH]cc(C)c(=O)c2)=O)CN(C(=O)C(C)n2cccn2)C2(CCC2)C1 c1(CC(=O)NC2(c3nn[nH]n3)CC2)ccc(CC(C(F)(F)F)N2CCCCC2)cc1 C1(CNC(C2CC3(C2)CC32CC2)=O)CC2CN(C(c3cncnc3)=O)CC12 C1(NC(c2c(CC)nns2)=O)CN(C(C2C3CNC(=O)C23)=O)CC1CC(C)(C)C c1(C(=O)NCC2(NC(COC)=O)CCCCC2C)cnc(C(F)(F)F)c(C#N)c1 C(C(=O)NCCCCC(=O)NC(c1cscn1)CO)(C(C)C)OC c1(NC(c2c(COC)nn(C)c2)=O)ccc(NC(=O)C(C)(C)CN(C)C)c(C)c1 N1(C(CC=CC)=O)CCCCC1CC(=O)N(CC)CC1(C#N)CC1 C(CCC(O)C(=O)NCC1CCC(F)(F)C1)NC(C1C(C)(C)C1(F)F)=O Cc1nc(C(N2CCC2CNC(C2CC23CC3)=O)=O)cn1C c1(C(N2CC(CS(C)=O)C2)=O)cccn2c(CO)nnc12 S(=O)(=O)(c1ccc(C)cc1F)NC1CCN(Cc2scc(C(=O)OC)n2)C1 C(=O)(C1=CC2(CCOCC2)C1)N1CC(OC)C(NC(c2nc(Cl)sc2C)=O)C1 C1(NC(C(c2cccc(O)n2)C)=O)CCCCCN(C(C2CC2OC(C)(C)C)=O)C1 C(CC(CC)C(=O)NCC(O)CN(C(=O)CN(C1CCSC1)C)C)=CC N(C(=NCCSC(F)F)NCC(C)CN1CCCCC1)C1C(C)C1 c1(O)ccc2c(c1)OCO2.C(C(=O)NC(c1ccccc1)C)(C(C)C)NC(C)=O c1(OC)cccc(OC)c1CC(N1CC2CC1C2NC(C1(C)CNC(=O)C1)=O)=O CCC(C)CC(C(=O)Nc1cnc(CC)nc1)NC(=O)Cc1cnc(C)s1 C(=O)(C=CS(C)(=O)=O)NCC(C(C)C)NC(=O)Cc1ccccc1Cl c1(C(N2C(CN(C(CCOCC(C)C)=O)C)CCC2)=O)cccnc1S N1(C(CCC=CC)=O)CCCC2CN(C(c3ccc(F)cc3O)=O)CCCC12 N1(C(Cc2ccc(C)o2)=O)CCC2(C=C(C(=O)NC(c3ncnn3C)C)C2)C1 C1(C(=O)NCC(CC)(C)Cl)CN(C(=O)Cn2cnnn2)CC12CCC2 N1(C(CCOC(C)=O)=O)CC(NC(c2cnc(O)n(C)c2=O)=O)C(C2CC2)C1 c1(CN2CC(C(C)C)OCC2)ccc2c(c1)CCN(C(=O)C(C)(C)Br)C2 N1(C(Cn2c(C)cc(C)n2)=O)CCOCC(C(=O)NC(C2CCOCC2)CO)C1 C1(C(C)(C)C(=O)NCC(F)F)CCCN(C(=O)C(=O)NCCCn2cnnc2)C1 O=C(CC1CCCCc2ccccc21)NC(c1ccc(F)cc1Br)c1ccccc1 CC1C(C(=O)NC2CCN(C(N)=O)C2)CCN1C(=O)Cc1ccn(C)c1 C1(NC(CC2(C)CC2)=O)CN(C(=O)C=CS(C)=O)CC1c1ccc(F)cc1 c1(C(=O)OCC)ncc(N2CCC(NCC(C)O)CC2)nc1N c1(C(N(C(c2cn(-c3ccnc(F)c3)nn2)C)C)=O)ccc2c(c1)OCC2 N1(C(CC(C)SC)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)C(F)C(C)(C)O N1(C(CCC(=C)C)=O)CCC2CCC(NC(c3ccc(F)cc3N)=O)C12 C1(C(=O)OC)CN(C)C(=O)CN1C(=O)CC(C(F)(F)F)c1ccon1 C1C(CC(C)C)C(=O)N1.C1CCC(=O)N1.C(C)(CO)(C1CCC1)N.CCCOC(C)=O C1(CC(N2CC(N(C(c3n(CC)ncc3Cl)=O)C)C2)=O)CCCNC(=O)C1 C#CCC(C(=O)N1CC(C)(C(N2CC(C3CCCO3)C2)=O)C1)NC(C)=O C(=O)(C(CC1CCOCC1)NC(=O)CCC1(C)CC1)NC(C1CC(OCC)C1)=O c1(CC)cc(C(=O)NCC2CC(NC(=O)CCc3scnc3C)C2)ccc1C C=CCC(C(=O)N1CCCC1(C(=O)NCC(O)CC1CCCC1)C(C)C)OC C(=O)(CCCCCO)NC1CCC(CNC(CCC(C)SC)=O)C1 C(C(C(=O)N1CCCC(CCC)CC1)C(C)(C)C)NC(C(C(=C)C)(C)C)=O CC1(C)CC(n2nc(-c3cccc(F)c3)nc2-c2cccc(C(C)(F)F)n2)CO1 C1(F)(CNC(=O)CSCCC(F)(F)F)CCN(C(=O)COCCCF)C1 C1(NC(c2ccc3c(c2)CCCC3)=O)CC2CN(C(=O)CC3CC3)CCN2C1=O C1(C)(CNC(c2nn(C)c(CO)c2)=O)CN(C(C2(C)CC3CCC2O3)=O)CCO1 c1(C(=O)NC2CCN(C(c3c(Cl)ncc(C)c3)=O)C2)c[nH]c2cc(F)c(F)cc12 C12(C(=O)NCC(C)NC(Cc3c(C)ocn3)=O)CCCCCC1OCC2 C1(C(N(C)CC2(CNC(c3cocn3)=O)CC(F)(F)C2)=O)Cc2ccccc2C1 C(=O)(C(C)(C)CC(=O)N1CCC(N(C(=O)CC2(O)CCCN(C)C2)C)C1)OCC N1(C(C(CC#C)C)=O)CC2(CCCC(CNC(c3cc([N+](=O)[O-])c[nH]3)=O)O2)C1 CC(C)C(F)(CNC(=O)CC1CSC1)C(=O)N1CCC(C)OC(C)C1 N1(CC(CC)C)CCCC(C(=O)Nc2csc(C)n2)C1 C12(NC(CSC)=O)CCN(C(c3cccc(N)c3Br)=O)CC1C2 N1(C(c2c(C)cc(Br)cc2)=O)CC2CCN(Cc3c[nH]ccc3=N)CC12 CCCCCC(O)C(=O)NCCN(C)C(c1cccc(C2CNC(=O)C2)c1)=O Cc1cn2c(n1)CC(C(=O)NC1CC(CNC(C3(C)CCCCNC3=O)=O)C1)C2 C1(C(N(CCCCCNC(C=C(C)C)=O)C)=O)CCCC12CC2 C1(O)(c2cn(C(CC)C)nn2)CCN(C(c2ccc(CN(C)C)c(F)c2)=O)CC1 c1(CNC(c2n(CC)ccn2)=O)ccc(C(=O)N(C2CCCC2C#N)C)nc1 c1(CC)oncc1C(c1nnnn1CC(F)F)NCc1ccns1 C(=O)(CC1=NN(C)C(=O)C1)NCCC(C)NC(C1CCCC(=O)CC1)=O c1(C(=O)NC2CC(C)(CNC(C=C(C)C)=O)C2)ccnc(Br)c1N C1(n2c(-c3cc(Cl)c[nH]3)nc(CCCC)n2)CC(C)(C)OC1(C)C N1(C(CCC(=C)Br)=O)CC2CC(C)N(C(=O)C3=CC(C)(C)C3)C2C1 C1(CC)C(NC(C2COCCC2(F)F)=O)CCCN1C(c1sccc1C)=O c1(C(=O)NC2CC(NC(C(C)NC(CC)=O)=O)C2)cncc(-n2ccnc2)n1 CC1CN(C(=O)C=C2CCC2)C(C)CN1C(c1cccc(OC(F)F)c1)=O c1(N2CC=CC(NC(=O)COCC3CCOC3)C2)ncc2ccsc2n1 C1(C(=O)NCc2cccc(OC)c2)CCCCCCN1C(=O)C(C(C)C)NC=O c1(C(=O)NC2CCC(N(C(COC)=O)C)CC2)cc2c(nc1N)CCCC2 c1(NC(C(C)(C)N)=O)ccnc(N2CCCC2)c1 C=CC1(C(=O)NCCn2cnnc2)CCN(C(C2CCC2C#N)=O)CC1 C(=O)(C1=NN(CCO)C(=O)CC1)N1CCC(F)(CNC(C23CC(F)(C2)C3)=O)C1 c1(C(=O)NC2C(NC(c3ccc(=N)[nH]c3)=O)CCC2)cc2cc(F)cc(F)c2[nH]1 C=CCC(CNC(C1C(O)CCN1C(c1c[nH]cc1CC)=O)=O)CC(C)C C1(OC)CN(S(=O)(=O)N(C)CCNC2CCCNCC2)CC12CCCC2 Cc1ccc(Br)cc1C(=O)NCC1CCCCN1C(C1CCC(=O)O1)=O Cn1cc(C(N2CCOC(CCNC(=O)C(F)=CC3CC3)C2)=O)c(O)n1 c1(C(N2CC(COC)N(C(=O)C(C)CN(C)C)CC2)=O)ccc2cncn2c1C c1(NC(C(C2CC(C)OC(C)C2)F)=O)cc(F)c(N)c(F)c1F c1(N(CCNC(c2cccc(CC)n2)=O)CC)ncnc2cc(C)[nH]c12 c1(SCC(=O)NC(CNC(C(C)OCCC=C)=O)C2CCC2)ccc(O)cc1 c1(C(N2CC3(C(C(N4CC(OCCF)C4)=O)C3)C2)=O)cc(F)ccc1Br CC(CN(C)C)C(=O)NC(CNC(c1conc1C1CCC1)=O)C1CC1 c1(C(N(CCCNC(c2c(COC)nn(C)c2)=O)C(C)C)=O)cccc(N)c1C c1(C(C(=O)N2CCC2CNC(=O)C=CC2CCOC2)OC)ccc(F)cc1 c1(CN(C(=O)CCOCCCNC(c2ccccc2F)=O)C)cccnc1O c1(SC(=O)CN2CC(C3CCCN3Cc3nnc(C)o3)C2)cccc(C(N)=O)c1 c1(N(C2CCN(C(C3CCCO3)=O)C2)C(=O)COCCO)ccncc1C(F)(F)F c1(C(=O)NCCCCN(C(=O)CC2(C#N)CCCCC2)C)c(Cl)cccc1[N+](=O)[O-] C1(O)(CC#C)CC(C(=O)NCC#CC(=O)NCCCC=CC)C1 C1(CC)CN(C(=O)CCc2cn(C)cn2)CC1NC(=O)CC1CC2CC2C1 c1(CNC(C(C)(C)OC)=O)c[nH]c2ccc(I)cc12.C12CCCN1C2=O CC1CN(C(C2C=CCN2C(=O)C(O)CC2CCCC2)=O)CC(C)(C)CO1 Cc1cc(C)c(NC(=O)C(N2CC(C)C(F)(F)C2)c2cn(C)cn2)c(C)c1 c1(CC)noc(C(=O)NC(C)(CNC(c2ccc(OC)nc2)=O)C2CCC2)c1C C1(CC)CN(C(=O)C(C2CC2)SC)CC1C(N1CC(COC)(OC)C1)=O C1(NC(C(C)OCC#C)=O)CC2(CCC(NC(C3(C4CCC4)CC3)=O)CC2)C1 C1(C(=O)OC)(CN2CCN(C(=O)NCCOCCF)CC2)CCCNC1 N1(C(C=C(C)Cl)=O)CC2CC1CC2CNC(=O)CCC1CCC(C(F)(F)F)CC1 C(=O)(CS(=O)(=O)C1CC1)NC1CC(C(C(N2CC(C)C(N(C)C)CC2)=O)F)C1 Cc1cc(C(N2CCN(C(c3ncoc3C3CC3)=O)C(CF)C2)=O)cc(N)c1 N1(C(C2CCS2(=O)=O)=O)CCCC1C(=O)N(CC(O)CO)CCO C1(CN(C(C2CCC(C)C2)=O)C)CCCCN1C(c1coc(Br)c1)=O N(C(=NCc1ccccc1)NCC1CCN(CC(F)(F)F)C1)CC(CC)CO c1(CNC(C2C(c3onc(COC)n3)(C)C2)=O)nccc(O)n1 N1(C(CSC(C)C)=O)CCC(C(C)NC(=O)Cc2cc[nH]n2)CC1 C1(CNC(CNC(CC)=O)=O)CN(C(=O)C(C)SC)CCC1(C)C C1(NC(C(C(C)O)N(C)C)=O)CC2CCC(C1)N2C(c1sccc1C#N)=O N1(C(C2CN(C(=O)NC)C2)=O)CCCN(C(=O)C(F)N2CCCC2)CC1 C(=O)(C(O)CC(C)(C)C)NC(=O)Oc1cccc(OCCNC(=O)NC)c1 C1(C(N2CCN(C(=O)CCC3CCCCN3C)CC2)=O)(OC)CCSCC1 c1(C(=O)NC2CC3C(NC(c4cnc(OC)s4)=O)C3C2)cc(F)c(C)cc1N N1(C(C(COC)O)=O)CC2CCC1C1CN(C(c3cnn[nH]3)=O)CC21 N1(C(C2CC(=C)C2)=O)CCC2(CCCCC2NC(c2nc(C(C)C)oc2C)=O)C1 c1(C(N(C2CN(C(Cc3ccc(C)s3)=O)C2)C)=O)ccc2c(c1)C(C)CN2 c1(C(=O)NCC2CC(NC(c3nccnc3Br)=O)C2)ccc(CO)c(Cl)c1 c1(C(=O)NC2CN(C(c3cc(OC)n[nH]3)=O)CC(O)C2)n[nH]c2c1CCCCC2 C1(NC(Cc2ccc(C)cc2)=O)CCN(C(C2CC=CCO2)=O)CC12CCC2 c1(OCC)cc(Cl)ccc1C(N1CC2CC2(NC(C2C=CCC2)=O)C1)=O c1(OC)cc(Cl)ccc1-c1nccn1N(CC)Cc1ccc(C2CCC2)cn1.C(C)C C#CCC(C)C(=O)N1CCC(NC(c2c(C)nsc2NC2CCCC2)=O)C1 C1(C(=O)NC2CN(C(=O)CCF)C2)CC(=O)N(C2CCCCCC2)C1 C(c1ccc(F)c(F)c1)=CC(=O)Nc1ccc(NCC(C)(C)C)cc1 N1(C(C(F)=C(C)C)=O)CC2(C1)CN(C(C1CC1c1cn[nH]c1)=O)CC2CO c1(CN(C2(n3cc(C(=O)O)cn3)CC2)C)conc1C(C)(C)C Cc1ccccc1C(C)(C)C(=O)NCC1CC(NC(=O)CSCC(C)C)C1 CN=c1nc(N2CCC(c3cc(=N)[nH][nH]3)CC2)[nH]c(=NCc2csnn2)[nH]1 c1(C(N2CCOCC2)CNC(c2csc(C(F)F)n2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NC2CN(CC3C(OC)CC3)C2)nccc(Cl)c1O.c12ccc(cc1)CO2 CC(C)(C#CC(=O)NC1CCCC(O)CC1)CNC(=O)CCCN1CCCC1 C(CC(C)C(=O)NCC(C1CCC1)NC(=O)CCc1c[nH]c(C)c1C(C)=O)=CC c1(NCC(c2nccs2)C)nc(N(C)CC2CCOC2)nc2c1ncn2C Cc1cc(C(=O)NCCC(C)(C)NC(c2nnc(S)n2C)=O)ccc1C(F)(F)F Cc1ccc([N+](=O)[O-])c(C=CC(=O)NCC(O)CN(C)C(c2coc(Cl)c2)=O)c1 C1(NC(=O)COC2CCN(C(c3cn[nH]c3)=O)C2)CCC2(CCC2)C1 N1(C(C2C(C(C)C)C2)=O)CC(C(=O)NOCC(C)O)CC12CCC2 C1(CC)CCOCCN1C(C1CCNCC1)=O C1(C(=O)NCCN(C(C2(C#N)CC3C=CC2C3)=O)CC)CCn2c(cnc2C)C1 c1(C(=O)NCCC2(O)CN(C(=O)Cc3cscn3)C2)cnc2c(c1)C(=O)NC2 C(=O)(C(C)CCC(C)(C)C)N1C(CNC(C=CC(CC)=CC)=O)COCC1 C1(C(N2CC3C(CNC(c4c(C)nccc4Cl)=O)(C3)C2)=O)CC2(CCCC2)CO1 c1(C(N2CCN(C(C3(C(=C)F)CCC3)=O)C(C)C2)=O)nnn2cc(C)nc(O)c12 Cc1ccn2ncc(C(=O)NCC(C)(O)CNC(c3ccc(C)c(Cl)c3)=O)c2c1 c1(CC(=O)NC23CC2CNC3=O)ccc(CF)cc1.Cn1ncnc1CO c1(C(N2CCCCC2NC(=O)OC(C)(C)C)C(=O)NCC)ccc(C)c(C)c1C Cc1cc(Br)ccc1CC(N1CCC(CNC(=O)Cc2ccon2)C1)=O c1(NCCCCCCCC)ncccc1S(=O)(=O)NCc1nc(=N)n(C)[nH]1 c1(N(CC)CC2CCN(C(c3c(C)csc3Cl)=O)CC2)ccc2c[nH]nc2c1 C1(C)(CNC(CN(CC)CC)=O)CCN(C(C23CCCC2(C(N)=O)C3)=O)C1 c1(OC)cc(Br)ccc1C1CC1C(=O)NC1CS(=O)(=O)CC1N C(=O)(C(C)(C)C(N)=O)N.C(C(=O)N(CCN(C)C)CCCCN)N(C)CCOCCO N1(C(c2ccc(C3CCCO3)cc2)=O)CCCC(C2(O)CC2)C1 N1(C(=O)CCn2ccnc2)CCC2(CCCN2C(c2ccccc2CO)=O)C1 Cc1cc(O)cc(C)c1C(=O)NCC12CC(NC(=O)CCCCC(F)F)(C1)C2 C1(CNC(C2(C)COC(=O)C2)=O)CN(C(=O)CCc2ccoc2)C(C)(C)C1 C1(O)(CCNC(=O)CCC2CCC2)CCN(C(C2CCN(CCF)CC2)=O)CC1 N1(C(C(N2CCN(C(=O)CN3CCCC3)CC2)C)=O)CC2CCCC1CCC2 C(CNC(c1ncc(C)cn1)=O)(CC(F)(F)F)NC(CCC(=C)Cl)=O N1(CC)CC(C(=O)NCc2[nH]ccc2C(N2CC(c3nncn3C)C2)=O)CC1=O C(N=c1[nH]c(=NCCc2conc2Br)c2[nH]ccc2[nH]1)c1c(SC)ccnc1 N1(C(CCC2C(C)C2)=O)CC(CNC(=O)CC2(N(C)C)CC2)C2(CCC2)C1 Cn1c(O)nc(N2CC3C(C(=O)NCC45CC=CCN4CCC5)C3C2)cc1=O c1(N(C(=O)CC(N)CC2CCCN2C(=O)OC(C)(C)C)C)cc(F)cc(Cl)c1 N1(C(CC2N(C(C(CCC(C)C)=O)=O)CC3(CC3)C2)=O)CCC(C)C2(CCC2)C1 N12CCC(CC1)NC2=O.c1(SC(C)C)ncc(C(=O)OC(C)(C)C)s1 C1(CNC(C2(N(C)C)CC2)=O)C2CN(C(=O)C(O)C3CCCC3)CC12 N1(C(CC2CN(C(COC)=O)CC23CC3)=O)CC2(CNC(=O)N2C)C1 N1(C(c2c(C)nn[nH]2)=O)CC(C2CN(C(c3cc(Cl)nn3C)=O)C2)C1 Cc1ccc(C(=O)NCC2(NC(=O)CC(O)C(C)C)CC2)c(Cl)c1Cl Cc1ccc(F)c2oc(C(=O)NC3CCC(NC(c4cscc4F)=O)C3)cc12 Cn1nnc(C(=O)NCCC2CC(NC(=O)C(O)C3CCCC3)C2)c1C(F)(F)F c1(CN(C(C2(CNC(=O)C(=O)Nc3ncc[nH]3)CCCC2)=O)CC)ccccn1 C1(O)(C(=O)NCCN(CC2CC2)OC2CCOC2)CCOC1.O=c1ccc1=O CC1=C(C(=O)NC2CN(C(c3ccc(C)nc3C)=O)CC2(C)C)CCC1 N1(C(c2cc(C(=O)OCC)ncc2)=O)CCCC(C)(COCC#N)C1 c1(C(C(=O)OC)NCC2(CO)CC(F)(F)C2)ccc([N+](=O)[O-])cc1 N1(C(CCC#C)=O)CC(CNC(c2cccc(N(C)C)n2)=O)OC2(CCC2)C1 Cc1nnc2n1CC(C(N1CC(C)(C)OC(C)(C)C1)=O)N(C(c1cscn1)=O)C2 C1(CC(N2CC(C)(OCC)C2)=O)CC(C)N(C(C2CCC(O)C2)=O)C1 c1(CC(C(c2nnnn2C)Nc2cc(CCCC)ncc2)C)ccc(F)cc1F CC1CCN(C(C2(C(=O)N(C)C)CC2)=O)CC1CNC(=O)CC1CCCCC1O c1(C(N(C(C)CCNC(C2CCC=CCC2)=O)C)=O)cnc2[nH]c(=N)sc2c1 C1(CCC)(NC(=O)C(O)C(C)C)CCN(C(=O)CC2CC2C)CC1 C(=O)(C(C)S(N)(=O)=O)Nn1cc(C2N(c3cc(COC)ncn3)CCCC2)nn1 C1(C(=O)NCC(C)(C)CO)CC2CCC1N2C(=O)Cn1cc(Cl)cn1 c1(C(N2CC(C(C(=O)NCC3(O)CCC(C)C3)O)C2)=O)ccc(O)cc1F C(CCCC(=O)NC(C1CC1(F)C(=O)OC)=O)NC(CNC)C C(CCC(=O)NCC1C(NC(=O)CNC(C2CCCOC2)=O)C1(C)C)=CC c1(CN(CCc2ccc(NS(=O)(=O)CC3CCCC3)cc2)CC)ccc(Br)c(Cl)c1 c1(C(N2CC(CNC(C3C(C)OCC3)=O)C2)=O)cccc2c1OC(F)(F)O2 c1(CCC(=O)N(CCNC(C2(C)CC(=C)C2)=O)C)c(C)ncnc1O CC(N=c1[nH]c(=NC2CCC(CO)CC2)[nH]c2ccsc12)c1ccc(F)c(Cl)c1 N#Cc1cc(C(N2CC(C(=O)Nc3cc(F)cnc3Br)C2)=O)ccc1O c1(OC)ccc(SC)c(OC)c1C(N1CCC(NC(=O)CCCCCOC)C1)=O N1(C(CCC(C)OCC)=O)CCC(C)(NC(=O)CCn2ccc(O)nc2=O)CC1 [N+]1([O-])(C(=O)CC2(C3N(C(=O)Cc4nnc(O)s4)CCCC3)CC2)CCCS1(=O)=O C1(CC)(NC(C2COCCC2(F)F)=O)CCCN(C(c2cnn3c2CCC3)=O)C1 c1(C(=O)NC2CC(C)CN(C(=O)C=C3CCCCC3)C2)nccc2c1CNC2=O c1(CC(=O)NC2C(NC(C=CC=CC)=O)C2)ccc(NC(=O)CNC(C)=O)cc1 C1(C)(OC)CN(CC(=O)NC(C)CNC(=O)Cc2csc(-c3ccsc3)n2)C1 CCC(C)(COC)C(=O)NC1CCN(CCCNC(=O)Cc2ccoc2C)C1 c1(NC(C2CC3(C2)CN(C(=O)CCc2cncnc2)C3)=O)ccc(Cl)c(F)c1 C1(NC(CSSC)=O)CN(c2nc(Cl)ncc2Br)CC(C)(C)C1 C=CC1COCC1NC(C1CC(NC(C2(CC)CCCCC2)=O)CCO1)=O Cc1c(CNC(C2(NC(=O)CC(=O)OC(C)(C)C)CCCC2)=O)cnn1C C(CCC(C)(C)C(=O)N(C1CN(C(C)=O)C1)C)NC(C(C(=O)OC)C)=O C(=O)(CN=c1[nH]c(C)cs1)N(CCCCN(C(C=CC=CCC)=O)C)C N1(C(CN(C(C)=O)C)=O)CCC(C2CC2)C1CNC(c1ccc(Cl)nc1Cl)=O c1(C(CNC(CC2(C=C)CC2)=O)NC(=O)CSc2cnn(C)c2)cccc(Cl)c1Cl N1(C(=O)COC(F)F)CC2CS(=O)(=O)CC2(NC(C2(F)CCCCCC2)=O)C1 Cc1nc(F)ccc1C1CN(c2cnc(Cl)[nH]c2=N)C1 c1(NC2(CNC(C3C(CC)OCC3)=O)CCOCC2)ncc2ncn(C)c2n1 C(C)(CCC=C(C)C)(c1n(C(C(=O)OC)C)nnn1)NCC1CC1c1cncs1 c1(C(N(C2CC(NC(c3ccc(N)cc3O)=O)C2)C)=O)cccc2c1CCC2 C(c1ccccc1)=C(C)C(=O)NC1CC(O)C1.C12CC1CN(C)C2=O c1(C(C(=O)NC(CNC(c2c(C(N)=O)cccc2)=O)CO)O)ccc(F)c(Cl)c1 C1(F)(CNC(C(COCC)C)=O)CCN(C(C2(N(C)C)CCOCC2)=O)C1 C1(CCC=C)(C(=O)NC(c2ccnn2C)C)CN(C(=O)C=CC=CC)C1 C(C(=O)NOCC1(C)CC1)(C(C)(C)C)NC(C(C1CC1)OC)=O C(=O)(C(C)(F)C(=O)N1CCN(C(C)CNC(=O)C(C)(C)SC)CC1)OCC c1(Cn2c(N(CC)CC3CCC3)nnc2-c2ccc(C)s2)c(C)nn(C)c1C Cc1nc(CC(N2CC(O)(CNC(c3cnoc3C)=O)C2)=O)n[nH]1 c1(NC(=O)Cc2ccnc(O)c2)cnc(SCCN2CCOCC2)nc1 c1cccc(N=S2(=O)CCCC2)c1.Cc1nc(C2CCOCC2)ncc1 c1(NC2CC(CNc3c(OCCOC)cncn3)C2)c[nH]c2nc(CO)ccc12.OC CC(CC(=O)NCC(F)CNC(=O)CCSCC(N)=O)c1cnn(C)c1 C#CCCN=c1scc(-c2sccc2Cl)n1CCC1CCC(F)(F)C1 C1(CNC(C23CCC(CC2)OC3)=O)CC2(C1)CC21CC1.C12(CC1)C(=O)N2 N1(C(c2[nH]cc(C)c2)=O)CCN(C(=O)CSc2n[nH]c(C)n2)C2COCC12 C1(NC(c2cncc(C)c2)=O)CC(C(=O)N(C)CC2CCSC2)=CC1O C(=O)(C1=NOCC1)NC1C(NC(CNC(C2CCCC2)=O)=O)CC1 c1(C(=O)NC(CC(F)(F)F)c2ccc(C(F)(F)F)cc2)cc(I)cc(Br)c1C c1(C(N(CCCN(C(Cc2n(CC)cnn2)=O)C)C2CC2)=O)ccc(SC)cc1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCC2(C1)CN(C(=O)CNS(C)(=O)=O)CC(C)O2 CC(C)CC(C)(C)C(=O)NCC(F)CNC(c1cc2ccccn2c1)=O C1(CCNC(C=CCN(CC)CC)=O)CCN(C(c2cc(C)oc2C)=O)C(C)C1 Cn1ncc(S(N)(=O)=O)c1C(=O)NCCN(C(=O)CSCc1ccccc1)CCF C1(CNC(c2cncc(OC(C)(C)C)c2)=O)CCN(C(=O)CC2CCCO2)C12CC2 N1(C(C2CCCCCC2(F)F)=O)C2COCC1CC(F)C2 C12(C(=O)NC3CC4CN(C(C5CN(CC)C(=O)N5)=O)CC43)CCC(CC1)C2(C)C N1(C(C(C2(O)CCCCC2)N(C(CN2CC(C)(C)C2)=O)CC)=O)Cc2ncsc2C1 Cc1nn(C)c(C)c1C(N1CCC1CNC(=O)C(O)CN1CCCC1)=O c1(NC(C)=O)ccc(C(=O)NC2CCCC2NC(c2ccc(C(N)=O)s2)=O)cn1 C(=O)(C1CCCc2scnc21)NCC(C)(C)NC(c1cccc(CCC)c1)=O N(C(=NCC)NCC1CCCC(C)O1)CC(C=C)(F)F c1(C(=O)NCC(C(=O)N(C(C)C(C)SC)C)OC)ccnnc1O O=C(CC(C(F)(F)F)c1nccn1C)NC12CC(C1)N(C(C1CC1(F)F)=O)C2 CCN=c1[nH]c(C)c(C(=O)NC2CN(C(c3cc(C)nc(O)n3)=O)CC2C)s1 CCC(CCC(=O)NCc1cc(C(N2CCCC2C2CCCC2)=O)ccn1)OC Cc1ccc(F)cc1NC(C1CCC(C)CN1C(=O)C(C)C(F)F)=O N1(C(C2C(=C)C2)=O)CCOC2(CCN(C(c3cc(Cl)cc(Cl)c3Cl)=O)C2)C1 C(=O)(CCC(C)(C)F)NC1CC(CC(=O)NCC2(OC)CCCCC2)C1(C)C c1(C(=O)NC2C(NC(Cc3c(C)noc3Cl)=O)C2)cccc(Cl)c1O CC1(NC(=O)CNC(=O)CC2CCCC2)CCC(C(=O)Nc2cn[nH]c2)CC1 N1(C(c2c(C)[nH]nc2Cl)=O)CC(NC(c2sc(C3CC3)nc2C)=O)C2(CC2)C1 c1(OC)cccc(C(=O)NCC(c2ccccc2)CNC(=O)CC(C)C)c1F S(=O)(=O)(c1ccc(C)c(Cl)c1)N(C1CCC1)CC1CCCN(C(C)=O)C1 C1(C(N2CC(OCC)C(CNC(=O)C(F)=C(C)C)C2)=O)CC2CCC1CC2 Cc1cc(C(=O)NCC2CC2NC(=O)C(C)CC(C)C)cc2ccoc12 N1(C(C(CSC)OC)=O)CC2(C1)CN(C(c1cccc(F)c1Br)=O)C2 CC(CNC(=O)CN1CCSCC1)CC(=O)NCCC(O)C(F)F O=C(CCC(=O)N1CCN(C2CCN(C(=O)CN3CC3)CC2)CC1)NC1CC1 c1(-c2cnc(CC)nc2)ccnc(Cl)c1OC.c12ccc(cc1)C(C)N2 c1(C(=O)NCC2CC(C(=O)Nc3cccc(CO)c3)CO2)cc[nH]c2nccc1-2 N1(C(CC2C(CNC(CC(=O)OCC)=O)C2)=O)CC(C)(C)C2CCCC12 C(=O)(CCCC(C)(F)F)NCCC(C)NC(=O)Cc1cnccn1 CC1OC2(C)CC1(C(N1CC(NC(c3cccc(F)c3)=O)C(O)C1)=O)C2 C1(OC)CC2CC(C(=O)NC3CCC(NC(c4cc(CO)ccn4)=O)CC3)CC12 c1(C(=O)NC2C(CNC(C(C)OC)=O)CCCC2)ccc2c(c1)CCCC2=O N1(C(CC(C=C)(C)O)=O)CCCN(C(C23CCC(C2)OC3C)=O)CCC1 C1(NC(C(C)=C(CC)C)=O)(CNC(c2ccnnc2)=O)CCC(F)(F)CC1 c1(C(=O)NC(CCCCNC(c2c(CC)[nH]nc2Cl)=O)C)ccn2nccc2n1 C12(CNC(CC(C=C)C)=O)CCCC(CN1C(=O)CCC=CC)C2 c1(C(=O)NCC2C3CN(C(c4cnc(F)c(Cl)c4)=O)CC23)cccc2oncc12 n1(CC)nc(C(=O)NC(C2CCN(C(C3(COC(C)=O)CC3)=O)CC2)C)cc1O CCCC(C(O)COC)OC(c1cc(C)n(C2CC2)n1)=O C1(CCNC(C(CC)OCC)=O)CSCCN1C(c1cc(C2CC2)on1)=O CON(CC1CCCCC1)C(=O)COCC1C2CCC(C2)C1C.C1CO1 N1(C(c2c(C)occ2)=O)CCN(C(=O)COC2CCOC2)CC2(C)CCCC12 C(c1sc(Cl)nc1Cl)=CC(=O)NC1CN(C(C2C3(CC3)C23CC3)=O)C1 c1(OC)cc(C(=O)NC2CCCC2(C)CC(C(=O)NC)OC)n(C)n1 c1(CNC(=O)NCC(c2ccc(F)cc2Cl)O)cnc2nccn2c1 c1(C(=O)NCC2CCC(NC(c3cc(C#N)on3)=O)CC2)c(F)cccc1Br C1(O)(CNC(=O)N(C2CC2)CC2CC2)CC2CCC1O2 c1(C(N2CCC(CC(=O)OC)C2)=O)cccc2c1CNCCO2 Cc1nc[nH]c1CC(=O)NC1CC(O)(CNC(=O)CCCSC(C)(C)C)C1 c1(C(CCC(=O)NCCCc2cc(Cl)sc2Cl)=O)ccc(Cl)cc1Cl N1(C(=O)Cc2ccc(F)cc2)CCCN(C(C2CCSC2)=O)CC1 N1(C(C2CCOC2=O)C(=O)NC)CCOCC1c1ncnn1C C1(NCCc2ccc(C)c(C)c2)CCCC(F)(F)CC1 c1(CC)nc(CNC(N2CCOC(c3ccco3)C2)=O)c(C)s1 C1(NC(CC=CC=C)=O)C2CN(C(C3CC4CC3C4)=O)CC12 CCCC(O)CC(=O)N1CC(NC(c2ccnc(O)c2Br)=O)CC(F)C1 c1(C(=O)NCCCN(C(C(C2CCOC2)OCC)=O)C)cc2n(n1)CCNC2=O N1(C(CC2OCCN(C(C3(C=C)CCC3)=O)C2)=O)CCC(CC)C(O)C1 c1(OC(C(=O)N(C(C)Cc2ccccc2C)CC#C)CC)ccc(C)cc1 C1(NC(C2CCC2C(F)(F)F)=O)CN(C(c2ccnn2CCF)=O)CC1C(F)F C1(NC(Cn2ccc(C)n2)=O)CC2(CCN(c3nncs3)CC2)C1 C#Cc1cc(C(N2CC(C(=O)NCC=CCSC)CC2(C)C)=O)ccc1C N1(C(C2CN(C(Cn3nnc(C)n3)=O)C(C)(C)C2)=O)CCOCC(C2CC2)C1 c1(C(N(CCNC(C2CCN(C(C)=O)CC2)=O)C)=O)nc(C)n2ccccc12 c1(OC)cc(C(=O)NC2COCCN(C(c3cnoc3C)=O)C2)c(F)cn1 C1(C(N2CCS(=N)(=O)CC2)=O)(NC(CC(C)(C)C2CC2)=O)CCC(C)(C)C1 CC(C)CC(CCO)NCc1ncccc1C(=O)O c1(NCCNC(c2n(C)nc(CC)c2Cl)=O)sc2cccc(F)c2c1C N1(C(COCCOC)=O)CCCC2(NC(=O)C=C3CC3)CC2C1 c1(C(C(N2C(C)CC(NC(CCC#C)=O)C2)=O)=O)cc(F)ccc1F c1(C(=O)NC(C(C)C)CNC(c2cn(C)nn2)=O)c(O)cnc2cc(F)ccc12 C1(CNC(CC)=O)CCCC2(CN(C(c3c(F)ccc(Cl)c3F)=O)C2)O1 C1(CC(C)NC(C2C(=C)CC2)=O)CCN(C(C2CCCC2(C)C)=O)CC1 C(C)(C(=O)NC(CNC(=O)CSCc1ccc(F)cc1)C(C)C)(C(C)C)OC Cn1c(=O)c2c(ncn2CC(=O)NC(C)(C)CC(F)F)n(C)c1=O N1(C(c2ccc(OC)nn2)=O)CCC(O)C(NC(c2ccccc2O)=O)C1 N1(C(COC(C)=O)=O)CCN(C)C(C(N2CCC(OC(C)C)CC2)=O)C1 N1(C(CC2C(C)OCC2)=O)CCC(C)(NC(c2ccnc(-n3ccnc3)c2)=O)C1 Cc1[nH]nc(C(=O)NC(CC2CCOCC2)C(=O)NC(c2cncs2)C)c1C N1(C(c2n[nH]c3c2CSCC3)=O)CCC2CCCCC12 CC(C)C(F)(F)CC(=O)NC1CC(CCNC(c2cnoc2-c2ccco2)=O)C1 C1(C(=O)NCC(N(C(CC)=O)C)C2CC2)CCCN(N2CCCC2)C1 N1(C(C(COCC)NC(c2cccc(CC=C)c2)=O)=O)CCC2(CSC2)C1 CC1CCC(NC(C2CCC(=O)N2C)=O)CN1C(c1cncc(N)c1)=O C1(C(=O)Nc2cccc(NC(C3(CCOC)CCC3)=O)c2)CCC2C1C2(F)F C(=O)(C1=CC2(CCOC2)C1)NCc1ccc(C(=O)NC(c2ccccn2)C)cn1 CC1=C(C(=O)NC2(C)CCCN(C(c3cncc(CO)c3)=O)C2)CCO1 C1(NC(c2c(C)nccc2)=O)CC2CCC1CN(C(=O)CCC1CCCCO1)C2 CC1CC(C(=O)NCC2(F)CC(CNC(C3CN(C)CCO3)=O)C2)=NO1 c1(C(N2CC(C(C(=O)NC(CO)CCCO)OC)C2)=O)ccc[n+]([O-])c1 C1(N(C(CC(CC)O)=O)C)CCC2CN(C(c3cnn(CC)c3C)=O)CC12 N1(C(c2cnc(OC)s2)=O)CC(O)CC1C(=O)NC1CCC12CCC2 C(C(C(=O)NOC1CC1)C(C)C)NC(c1c(C)ccnc1)=O C1(C(N2CC(C(C(=O)N(C(C#C)C3CCC3)C)OCC)C2)=O)CCC(=O)C1 c1(CN(C(c2sc(Cl)nc2C)C(=O)NCC(=C)C)C)ccc(O)cc1C C1(CC)CN(C(=O)CC2(C)CC2(Cl)Cl)CCN1C(=O)CC1CCN(C)CC1 c1(C(=O)NCCN(C(c2cscc2SC)=O)CC)cnc(OC)nc1 c1(C(=O)NC(C(=O)NCC(COC)C)CC2CC2)ccc2ccoc2c1 C1(C(=O)NC(CCC=C)(C)C)CCCCC1(C)NC(=O)CCC(=O)N(C)C1CC1 CCCC(C)(CCC)C(=O)NCC(C)(C1CC1)NC(c1cccc2nc[nH]c12)=O C#CCCCC(CCOC)NC(=O)CC(C)CNC(=O)CCOCCOCC C(C1CCCN1C(c1n[nH]cc1Cl)=O)=CC(=O)NCC(CO)C1CC1 N1(C(CC)=O)CCC2C(C1)CN2C(=O)C(C)C(O)CC c1(C(N2CCC(N(C(=O)COC3CCCCC3)C)C2)=O)cc(=O)n(C)cn1 C(=O)(CCCCc1ccc(F)cc1)NCC1(F)CC(NC(CSS(C)(=O)=O)=O)C1 C#Cc1cccc(C(N2CCC=CC2C(=O)NCC2CCCOCC2)=O)c1 C1(C(=O)NCCCC(=O)NC(C2CCCCC2)C)CC(C)CC(C)C1 C1(N(C(CC2C(C)CCC2)=O)C)CCC(NC(=O)CC(=O)NCC2CC2)CC1 C12CN(CCCO1)C2=O.n1(C2(C(=O)NCCCN(CCCC)C)CC2)nccn1 CCC(CC(=O)NCC1CC1C(N1CC(C(C)C)C1)=O)CC(C)C C1(CC(=O)N(C)C)CC(F)CN1C(=O)CC(=O)NC1CC1.c1(O)ccccc1 c1(C(=O)NC2(C)CN(C(C3CC4CCC4C3)=O)C2)nc2ccccn2c1F c1(C(=O)NC2CCN(C(C=Cc3c(C)cncc3)=O)C2)cc2cccc(O)c2[nH]1 Cc1ccc(=O)n(CC(=O)NCCCCCN(C)C(C23CCC2CC3)=O)n1 N1(CC(C2CCN(Cc3ccccc3)CC2)C)CCC(C2CC2)(CN)C1 Cc1cc(C)c(C(=O)NCC2CCN(C(=O)CCCN(C)C)C(C)C2)cn1 N1(C(c2c(F)ccc(CC)c2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC(CO)C1 N1(C(CC(=C=C)C)=O)CC2CC(NC(c3[nH][nH]c(=N)c3Br)=O)CC1C2 CCCCCC(O)C(=O)NC1CN(C(=O)COCC(C)C)C(C)(C)C1 c1(C(=O)NCC2CCCN2C(c2nncn2C2CC2)=O)c[nH]nc1-c1ccsc1 c1(C(N2CC(NC(C=CCC)=O)C(C)(C)C2)=O)cc2cccc(OC(C)=O)c2o1 c1(C(=O)NC2CN(Cc3ncc(OC)nc3)CC2F)n[nH]c2cccc(F)c12 CCCC(C(=O)NCC(O)CNC(c1ccc(Cl)cc1OC)=O)S(N)(=O)=O C=Cn1nccc1C(=O)NCc1ccsc1C(=O)NC1C(C)CCC1C C1(C(N2C3CC(C2)ONC3=O)=O)CC12CCOCC2.C=CC(C)NC(C)=O CC(CS(C)=O)C(=O)N1CC(CN(C(=O)CCC(Cl)Br)C)C1 Cc1ccc(NC(c2ccc(C(F)(F)F)s2)=O)c2ccccc12 c1(OC(C(N2C3CC(C(=O)OC)CC2CC3)=O)C(C)C)cc(C)cc(F)c1N c1(NC(c2cccc(NC(C3CCC(=O)NC3)=O)c2)=O)cc(O)cc(O)c1 C(=O)(CCC(C)(F)F)N1C(C(=O)NCC(C)(C)C2CCCO2)C=CC1 C1(NC(c2cnn(CC)n2)=O)CCN(C(c2ccc(C3CCC3)cc2)=O)CC1C C(C(C)(C)CNC(C1CCCC1NC(=O)Cc1cc(C)on1)=O)OCC C1(OCC)(CNC(=O)Cn2cc(C3CCCOCC3)nn2)CCS(=O)(=O)CC1 C#CCCCC(=O)NC1CCCN(C(c2n[nH]c(C)c2Br)=O)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NCCN(C(=O)CC1CCC(=O)NC1)C C#CC1(NC(=O)C=CC2CCCN2C(=O)C(F)C2CCC2)CC2CCCC12 C(CNC(c1c(CNC(c2cc(C3CC3)[nH]n2)=O)nnn1C)=O)(CC(C)C)OC C1(CN(C(=O)CC2CCC23CCC3)C)COCCN1C(c1cccc(CO)c1)=O c1(CCN(C)C)cnn(CC(=O)N(C2CCS(=N)N2)C)c1.C(CN1CC1)N.C(CO)O C1(c2ccc(SCC(C)Cn3ccnc3)cc2)CC12CC(F)(F)C2 C1(NC(=O)CCOC2CC2)CCC2(CCN(C(C3CCCC3C(F)F)=O)CC2)C1 C1(C(N(C(C)CNC(c2ccc(C(=O)OC)o2)=O)CC)=O)NC(=O)OC1C c1(OC)ccc(C(=O)NC2CCC2NC(=O)COCP(C)(C)=O)cc1OCCO c1(OC)cccc2cc(C(=O)NCC3CCN3C(C3(O)CCOCC3)=O)oc12 S(=O)(=O)(c1cccc(S(=O)(=O)N(C)Cc2ccc(C)cc2)c1)C1(CCCC)CC1 C=CC1(C(=O)NCC2(CC)CCOC2)CCN(C(=O)CCCC(=O)OC)C1 C12(C(N(CC#C)CC3CCCO3)=O)CC(CO)(CN1C(=O)C(C)(C)O)C2 CCC(C(=O)NC(C)(C)C(C)CC(=O)NC(c1cnn(C)c1)CO)C(F)(F)F C(=O)(C(C)CC(C)(C)C)N(C(C)C(=O)N(C)CCc1cnc[nH]1)CC c1(C(N2CC2=O)=O)cc(C)nc(C)c1.CCCCS(=O)(=O)NC(C)C C(=O)(C(N=[N+]=[N-])C(C)C)NCc1cc(C(=O)NC(C#CCC)(C)C)n[nH]1 C1(C(N2CCN(C(C)=O)CC2)C(=O)N(C(CC)C)C2CC2)CCCC1(C)C C(=O)(CC1=CCN(C)CC1)N1C(C(=O)NC2CCCN(CC)C2)CCCCCC1 C(=O)(C(C)C1OCCc2sccc21)NCC1(F)CC(NC(COC)=O)C1 c1(C(=O)NCC2C(NC(=O)C=CCO)CCC2)cncc2nc(O)[nH]c12 C1(C(N(CCC(=O)NC)C)=O)CN(C(c2cc(C)n(C)c2)=O)CCN1C C(=O)(C(CCC)C(C)C)N1CCN(C(C2CC3(CC(=C)C3)C2)=O)C2C1C2 C1(C)(COC)CC(C(F)(F)F)(OC)C1.C(CC(O)CC)n1cc(C)nn1 C1(NC(C2CC3(C2)CC3F)=O)CCCC2CN(C(C3(O)CCCCC3)=O)CC12 c1(C(=O)NC2CC(C)(NC(c3ccc(F)cc3Cl)=O)C2)cc(O)cc(C#N)c1 c1(NC(C2(C)CCCN2Cc2ncc(Br)cc2Cl)=O)cc(F)cc(F)c1[N+](=O)[O-] C1(C(=O)NC(COC)CCO)CN(C(=O)Cc2nonc2C)CC1(C)C N1(C(COC(CC)CC)=O)CC2C=CC1C(NC(C1CCCS1)=O)C2 c1(C(N2CCC(COC)(NC(C3CCC3)=O)C2)=O)c(C)nn(C)c1C C=CC1CN(C(c2c[nH]c(C)cc2=O)=O)CC1NC(=O)Cn1ncccc1=O NC12CC3CC(CC(C(=O)Nc4ccn5cc(CO)nc5c4)(C3)C1)C2 c1(OC)nc(NCC(C2CC2)NC(c2cc(C(F)(F)F)n[nH]2)=O)nc2[nH]cnc12 C1(CCNC(c2cnc(S)[nH]2)=O)CSCCN1C(=O)Cc1ccc(Br)cn1 Cc1c(C(=O)NCC2CN(C(C3CN(C4CCOC4)C3)=O)C2)ncn1C c1(C(=O)NC2CC3(CCC3)C2O)ccn2nccc2c1 CC12CCC(C(=O)NC3CCN(C(=O)CCNC(=O)OC(C)(C)C)C3)(C1)OC2 c1(OCCC)nc(C)ccc1C(=O)NCC(C)N(C)CC1C(C(=O)NC)C1 c1(CCC)nc(C(=O)NC(c2cn(C)nn2)C(=O)NC(C)Cc2ccco2)co1 c1(C(=O)NCCNC(c2ccc(OC)cc2)=O)cc(Cl)cc(F)c1N C(CCC(C(=O)NC1CC2(CCC2)C1O)NC(C12CCCC1C2(F)F)=O)OC O(NC(=O)C(NC(=O)C(C)C)SC)CC=CC.OC C=C=CCCC(=O)NCC(C1CCN(C(c2ccc(F)cc2)=O)CC1)(C)C c1(OCC=C)ccc(C(=O)NCC(C(C)(C)C)c2ccccc2)cc1 Cc1cn2cc(NC(N3CCN(C(=O)CSC(C)(C)C)CC3(C)C)=O)sc2n1 C(=O)(CCC(C)SC)NC1CCCC1CCNC(C1C(C(=O)OCC)C1)=O CN1CCOCC1C(=O)NCCCC1CCCCN1C(C1SCCS1)=O CC(CC(F)(F)F)N(CCC(=O)N(C)C)C(c1nnnn1C1CCCCCC1)C Cc1ccc(C(C)C(=O)N2CCC2)cc1.c1(CC=O)cccc(C)c1 N1(C(=O)NCc2cn(CC(C)NC(=O)Oc3ccccc3)nn2)CCCC(O)C1C N1(C(C(C(C)C)CNC(=O)CCCNC(N)=O)=O)CCCC(C2(C)CC2)C1 C(=O)(C(F)C(F)(F)F)NCCCN1CCN(C(C(CC)c2ccccc2)=O)CC1 C1(C(=O)NCC(C(C)(C)C)O)CCN(C(=O)Cn2ncn(C)c2=O)C(C)(C)C1 CC1C(C(=O)NCC(C)(C)CN(C(=O)CC(F)F)C)C1(F)F c1(N(CC(C)(Cc2ccccc2)CO)C2CCOCC2)ccc2c(c1)OCO2.C N12CC(C3(CC3)C1)CNC(=O)C1(CC1)C2=O.C1(NC(=O)OC)COC(C(F)(F)F)C1 N1(C(=O)CCc2cc[nH]n2)CCCCC1CCNC(C1CCCCC1)=O C(N=c1nc(N2CC3CC(C)(C)C3C2)c2sccc2[nH]1)C1(C)CCC(F)(F)C1 C12(C(=O)NCc3c(C)nns3)CCN(C(c3conc3C)=O)CCC1C2 N1(Cc2ncc(-c3ccc(C)cc3)c(C)c2)CCN(c2nnnn2C)C(C)C1C c1(C(N2CCC(NC(C(C)CC3CCC3)=O)C2C)=O)coc2c(F)cc(F)cc12 C=CCCCCCCC(=O)NCC(C(C)C(C)C)NC(c1ccc(C(C)=O)o1)=O N1(C(C(C=C)OC)=O)CC2CC(C(=O)Nc3ccccc3)C(C2)C1 C1(NC(C2(C=C)CC2)=O)CC12CCN(C(c1cc(CC)n(C)n1)=O)CC2 C=CCC(C)(CC)C(=O)NC(C)CC(C)NC(c1cncc(C(=O)OC)c1)=O C1(NC(c2c(C)snc2)=O)(CO)CCCN(C(c2cc(C(F)F)cc(F)c2)=O)C1 c1(C(N(CCn2cc(CCC3CC3)nn2)CC)=O)nc2cnccc2s1 N1(C(CN2CC(C)C2)=O)CCCCC1CCCNC(=O)C=Cc1cc[nH]n1 c1(CCCC(=O)NC2(CO)CC(C(C)(C)C)C2)c(F)cccc1F c1(C(N(C(C)C(=O)OC(C)(C)C)CC)=O)cnc2ccc(F)cc2c1 N1(C(Cc2c(C)cco2)=O)CCCC(C)C1CCNC(c1c(Cl)sc(C)c1C)=O C12(C(=O)NC3(CNC(C4CCOC4C4CC4)=O)CC3)CC=CC(C1)OC2 CN1CCC(F)(CNC(=O)CC2CCCN(C(=O)Cc3cnsc3)C2)C1 C1(N(C)C)CCCN(C(c2cn(CCNC(C3C=CCCC3)=O)cn2)=O)C1 CC(C)C(O)C(C)C(=O)N1CCCC(C(=O)NCCC2CCOC2C)C1C c1(OCC)cc(C(N2CCCC2C(C)(C)NC(=O)C=Cc2nccs2)=O)[nH]n1 C#CCC(CC(F)F)C(=O)NC(C1CCCN1C(C1CC(n2cnnc2)C1)=O)C1CC1 c1(CC)ccccc1C(=O)NCC1CCN1C(c1nc(C2CC2)cs1)=O C1(NC(C(C)OCC)=O)C2CC1N(C(=O)C=Cc1ccc(-c3ccccc3)s1)C2 N1(C(Cc2cn(C(C)C)nc2)=O)CCN(C(C23CC(F)C2C3)=O)CC(C)C1 n1(CC)cc(Br)c(C(=O)NCC(C2CC2)N(C)C(C2CC2CC)=O)n1 N1(C(c2nnn(CC)c2C)=O)CCC(NC(=O)CC(C)(O)C2CC2)C(F)C1 c1(C(N(C(C)CNC(=O)C=CC(N2CCC(C)C2)=O)CC)=O)ccn2ccnc2n1 c1(C(=O)O)ccc(Cl)c(S(=O)(=O)NCC2CC23CCCOC3)c1 CCC(C)C(O)C(=O)NC1CC(CNC(=O)CN2CCCCS2(=O)=O)C1 CCC(CO)CCNC(C1(CCNC(=O)CS(C)(=O)=O)CCCC1)=O Cc1cccc(C(=O)NC2C3CC2N(C(c2cnc(C4CC4)nc2)=O)C3)c1Br CC1(NC(=O)CC(CC2CC2)NC(C2(O)CCOC2)=O)CCCC1O N1(C(C2CC(C#C)(O)C2)=O)CCN(C(c2cnn(C)c2)=O)C(C(C)(C)C)C1 S(=O)(=O)(c1ccc(Br)cc1Br)N1CCC(C(=O)Nc2ccc(CCO)cc2)CC1 C1(C)(C(=O)NC2CN(C(COCCC(C)C)=O)C(CO)C2)CC(C2CC2)=NO1 Cc1cc(C(=O)NCC(=C2CN(C(=O)CC3CCC(C)CO3)C2)F)nc(C)c1 CCC(C)(CNCc1ccc(OC)cc1OCC(=O)O)C(C)O C1(C(=O)NCC(CNC(C(C)CN(C)C)=O)F)C2CCC3(COC(=O)C13)O2 CCCCC(CNC(C1CC(C(=O)OC(C)(C)C)C1)=O)NC(=O)COC1COC1 C(=O)(CCC(C)(F)F)N1C(C)(CNC(c2n(CCOC)ncc2)=O)CCC1 CC1CC(O)CN(C(C2CC2c2nc(-c3cccc(C(F)(F)F)c3)no2)=O)C1 C1(NC(=O)Cc2ccc(F)cc2)CCN(C(=O)Cc2csc(Br)c2)C12CC2 CCC(C(=O)N1CCC(C(=O)NC2COC3(CCC3)C2)C1)C(C)(C)CC C=Cn1nccc1C(N1CC(C(N)=O)(CNC(=O)CCOCCOC)C1)=O N1(C(C2(C=C)CCCC2)=O)CC2CC(NC(c3ncccc3Cl)=O)C1C2 c1(-c2cccc(CN(C(C(C(C)C)c3cccnc3)=O)C)c2)cn(C)ccc1=O c1(C(=O)NCCNC(CCC2C(C)C2)=O)ccc(F)c(S(=O)(=O)N2CCCC2)c1 N1(C(COC(C2C(C(C)(F)F)C2)=O)=O)Cc2ccccc2CCC1 C(=O)(C1=C(C#N)CCC1)NCC1(C(F)F)CCN(C(c2n(C)c(S)nc2)=O)C1 CC#CC1CCN(C(=O)OC2CN(CC(C)(C)C)C23CCC3)CC1 N1(C(c2n(C(C)C)ccn2)=O)CCCC2(C1)CN(C(=O)CN1CC(C)(C)C1)C2 c1(C(N(CC(CNC(COC(CC)C)=O)C)C)=O)cnc2cc(C)ccn12 CCC(CC(F)(F)F)C(=O)NCCCC(C)NC(c1nc(C2CC2)cs1)=O c1(CCCC)ccc(Cl)cc1C(=O)NC1CC2CC(NC(=O)CCC(C)C)C2C1 C(CCC(=O)NCCC1(C(=O)NCCn2ccnn2)CC1)N(C)C Cc1[nH]c(=NC2CN(C(c3c(Cl)nn(C)c3Cl)=O)C2)ccc1C#N N1(C(c2cc(C(=O)OC)n(C)c2)=O)CCN(C(=O)C(C)CSC)C(C2CC2)C1 N1(CCCNC(C(OCC)OCC)=O)CCN(C(=O)CC(=O)OC)CC1 c1(CC(=O)NC2C(NC(C34OC(C)(C)C(C3)C4)=O)CC2)ccc2c(c1)CCCO2 C1(C(=O)NCC2(CC)CCCO2)CN(C(=O)C(OC)OC)CC12CC2 C#Cc1ccc(CC(=O)NCC2CC2CNC(c2ncnn2C(C)C)=O)cc1 c1(NC(N2CCC(O)C2(C)c2ccccc2)=O)cc(F)c(F)cc1I C=CCC(C)(C)CC(=O)N1CC(N=[N+]=[N-])CC1C(=O)NC(C)C(C)F c1(C(=O)NC(C2CCOC2)CNC(CCC(=O)N(C)C)=O)ncc2[nH]ncc2n1 C=CC(C)(C)CC(=O)N1CC2(CC2)CC1CNC(C1CCC(F)(F)CO1)=O C(=O)(CC1OCc2ccccc21)NCCN(C(CCn1c(C)csc1=O)=O)C C1(CNC(CNC(CCC)=O)=O)(CO)CCCN(C(C2CC2CC)=O)C1 N1(C(CC(CCC)(C)C)=O)CC2CCC(C1)N(C(=O)CCc1nccs1)C2 O=C1NC(Cc2ccccn2)C(=O)N1c1ccc(CC2CCOC2)cc1 N1(CC(N2CCC(CNC(c3cn(CC)nc3)=O)C2)=O)C(=O)CSC1=S CCCCC(CC)CC(=O)NC(CCN(C)C(c1ncnn1C)=O)C(C)(C)C C1(CNC(CC=C)=O)CCC2(CCC2)C1NC(=O)CCN1CCC(C)CC1 c1(N2C(C)CC(NC(=O)CCc3cncnc3)C2)ccc(C#N)nc1 N1(C(C(CCN(C)C)O)=O)CC2CCC1C1CN(C(c3ccc(O)nn3)=O)CC21 c1(NC(C2C(NC(c3c(Br)cnc(Cl)c3F)=O)C2)=O)ncnc2[nH]c(Br)nc12 C1(NC(CC(C)C(F)F)=O)CCC2CCN(C(c3ncn4c3CCC4)=O)C12 N1(C(C(C)OCCCC)=O)CCC(NC(=O)CC2CC(=O)NC(=O)C2)C(C)C1 Cc1cc(F)cc2[nH]c(C(=O)NCC(F)CNC(=O)Cc3ccccc3)cc12 CCC(C)(CNC(=O)CN1CCCCC1=O)C(=O)Nc1cc(OC)ccc1C N1(C(CCCOC(C)=O)=O)Cc2n[nH]cc2C1C(=O)N(CC(C)F)C CCCC(C)(CC)C(=O)NCCC(C)CCNC(=O)C(C)NC(=O)Cn1cnnn1 CC1CN(C(C2CC(N3CCOCC3)C2)=O)CC1NC(=O)CCc1cccs1 C1(CN(C)C(c2cncc(N)n2)=O)CCCCN1C(=O)C(F)C1CCC1 N1(C(CN(C)CC)=O)CCC(O)(CCNC(=O)COCCc2cccc(F)c2)C1 CC(C)(C)CCCCCC(=O)NCC1CC(CCNC(=O)COC(F)(F)F)C1 N1(C(C(N2CCC(C)C2)=O)=O)CCCN(C(c2ccc3c(c2)COC3)=O)C(C)C1.C c1(NC(c2nc(NC(=O)C(=O)c3ccco3)sc2)=O)ccc2c[nH]nc2c1 C(CCC(O)C(=O)NCC1CCCO1)NC(CCC=C(C)C)=O N1(C(=O)C(F)c2ncco2)CCN(C(=O)C(O)C2CCCC2)CC2(CC2)C1 Cc1ccc(NC(=O)C(C)(CO)NC(=O)C(C)OCCN(C)C)cc1COC N1(C(C(C2CC2)OCC)=O)CC(OC)C(NC(=O)C(c2ccccc2C)(F)F)C1 C(CC(=O)N1CC(C)(C)CC1CO)(C(F)(F)F)NC(C1C(=C)C1)=O C1(NC(=O)Cn2cc(CO)nn2)COCCN(C(c2cnc(S)n2C2CC2)=O)C1 C12(CNC(C(C)OCC)=O)CC(CC)(CN1C(c1ccc(OC)cc1C)=O)C2 c1(C(=O)NC(C)(CNC(=O)CC2(C(F)(F)F)CC2)C2CC2)ncnc2ccsc12 CC1(O)COCCN(C(C2CCC=CC2NC(=O)CC2CC=CC2)=O)C1 Cc1cnnc(O)c1C(=O)NC1COCC1C(=O)NCCCOCC1CC1 c12ccc(Cl)nc1N2.c1(CNC(C2(C(F)(F)F)CC(=C)C2)=O)c(C)cccc1C N1(C(C(C)N(C(c2n(CC#C)cnn2)=O)CCC)=O)CCNC(=O)CC1 c1(C(=O)NCC23CC(CN2C(c2ccsc2Br)=O)C3)ccc2c(c1)NC(=O)CC2 N1(CCCCCNC(C(CC)OCCOC)=O)CCN(C(=O)CC(C)(F)F)CC1 Cc1nc2ncnn2cc1C(=O)NC1CC12CC(NC(c1cc(F)n(C)n1)=O)C2 c1(C(N2CCOC(C)C2C)=O)c[nH]c(=O)c2ccnn12 n1(CCC=C)nc(-c2ccncc2)nc1C1CCC1.n1(CC(C)C)nc(C)cc1C N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CCN(C(=O)CCc1ncc[nH]1)C2 c1(C(=O)NC(CN(C(C2CCOC2)=O)CC)C)ccc(Cl)c(N2CCNC2=O)c1 Cc1cc(-c2cn(C3CCN(C(C4CCS(=O)(=O)N4)=O)CC3)nn2)ccc1Br CC1CC(Nc2cc(COc3ccccc3)ncn2)C(C)O1 C#CCC(C)(CNC(C12CC(CO)(CN1C(C1CCCC(=O)CC1)=O)C2)=O)CO N1(C(COCCC)=O)CC(CNC(c2cccc(-n3cc(C)cn3)c2)=O)C(C)C1 N1(C(C(CC)C)=O)CCCC(C(=O)NC(CC)C(C)(C)O)C1CC N1(C(c2c(OC)nn(C)c2)=O)CC(NC(C23CC(F)C2C3)=O)C2(CC2)C1 N1(C(=O)NC)CCC(C(N2CCC(C(C)NC(C3CC(C)(F)C3)=O)C2)=O)C1 c1(C(N2CC(C#N)(C(C)C#N)C2)=O)cc2ccoc2cc1F c1(C(N2CCC(N(CCC)C(c3cocn3)=O)C2)=O)noc(CC)c1C Cc1cnc(C(=O)NCC2CC2C(=O)N(C)CCN(C)CCO)cn1 c1(CCC(N2CCC(OC(C=C(COC)C)=O)CC2)=O)ccc(C)c(OC)c1 c1(C(N(C(CC)CC(=O)N(CC(C)O)CC)C)=O)cccn2nccc12 c1(CC)nccc(C)n1.C(C)(CC(=O)NCC(=O)N(CC(=O)N(C)C)CC)=C(C)C c1(C(N2CC(CNC(C3(OC)CCC3)=O)C2)=O)ccncc1I C(=O)(C1=Cc2ccccc2C1)NC1C(CNC(=O)CCCc2cnn[nH]2)CCC1 N1(Cc2c(C)cc(Br)cc2)CCC2C(CCN2C(c2cncc(F)c2)=O)C1 c12ccc(nc1)SCC(C)O2.c1(NC(C=CC(=O)OCC)=O)ccccc1 C(=O)(C(CC)C(C)C)N1CCC(C(=O)NCCCC)(CC)C1 C1(C(N2CCCC(CCC(=O)NC3C(C)CCC3C)C2)=O)CC2(CCC2O)C1 N1(C(C(C=C)O)=O)CC(CNC(=O)CCc2ccn(C)n2)CC12CCC2 N1(c2ncccn2)CCN(C(C)CC2CC(=O)N(C3CCCCC3)C2)CC1=O Cc1cccc(-n2cc(C(=O)NC3CC(NC(c4cc(Br)n[nH]4)=O)C3)nn2)c1 N1(C(C(n2ncc(C)c2)C)=O)CC2CCCC(NC(=O)CC(F)(F)F)C2C1 N1(C(c2cnc(C(C)=O)s2)=O)CCC2CCN(C(=O)C(F)n3cccn3)C2C1 N1(C(C2=NNC(=O)C2)=O)CC2CC1CCC2NC(C1CCC(F)(F)C1)=O C1(C(N2C(CNC(c3cccc(O)n3)=O)CC2)=O)Cc2cncn2C(=O)N1 CCC(CC(=O)NCC1(CNC(C2(c3ccccc3C)CC2)=O)CCC1)SC CCC(C)(C(=O)NC1COCCN(C(=O)CCc2ncco2)C1)C(N)=O N1(C(C(C)c2ccsn2)=O)CC2CCN(C(c3csc4ccccc34)=O)C2C1 C1(CNC(CCCCC=C)=O)(NC(c2cc(C)oc2C)=O)Cc2ccccc2C1 C1(C(=O)NCC(CCNC(CCOCC#C)=O)O)CC2CCC(C1)C2(F)F N1(Cc2cn(Cc3ccc(OC)cc3)nn2)CCCCCCC1=O C(=O)(CS(=O)(=O)CC(C)C)NCC(CN(C(c1c(C)nc(O)cc1)=O)C)O N1(Cc2c(OC)nccc2)CCC2CN(C(c3occc3Br)=O)CC2C1 N#CC1(NC(c2cccnc2S)=O)CCN(S(=O)(=O)C(F)(F)F)C1 N1(C(C(C(C=C)C)C)=O)CCOC2(C1)CN(C(=O)CC1CC3(CCO1)CC3)C2 C1(C(N2CC(NC(C3OCC(CNC(COC)=O)C3)=O)C2)=O)CC12CC2(F)F C1(c2nnnn2CCC2CC2)(C(N(C)CCN(C)C)=O)CCOC1.C1(CC)CC1 c1(C(=O)NCC2CC(O)(CNC(CC3N(C)CCC3)=O)C2)nccc(Cl)c1F NS(=O)(=O)c1ccc(C(N2CCN(C(=O)C=C(Cl)Cl)C(CC(F)(F)F)C2)=O)o1 C#Cc1cccc(C(=O)N(C2CN(C(=O)Cn3cccnc3=O)CC2(C)C)C)c1 C(CCCC(C)NC(=O)CNC(N)=O)NC(C(C)OCc1ccccc1)=O CC(=NOCC#N)C(=O)NCCN(C1CCCC1)C(=O)CN(C1CCC1)C c1(C(=O)NCC2(C)OCCN(C(C(CC)=CC)=O)C2)cccc2ncnc(O)c12 C1(NC(Cc2cccc(NC(c3ccc(CC)s3)=O)c2)=O)CCCCCC1O C1(C(=O)NC(C2CCC2)C2CCC2)(CC)CN(C(C2CCC(C)O2)=O)C1 C1(NC(c2cc(C(=O)OC)oc2C)=O)C=CCN(C(C2CC2Br)=O)C1 C1(NC(C=CCOC)=O)CCC12CCN(C(c1cccc(C3CC3)c1)=O)CC2 C1(NC(C(CNC(C)=O)(C)C)=O)CCCN(C(=O)C(C)C2CCOC2)C1C C(=O)(CCS(C)(=O)=O)NCC(CNC(C12CCC(OC)C1C2)=O)OC c1(CC)ccccc1C(N1CCOC(CC(C)C)C1)=O.C1C(=O)NCCO1 N1(C(C(Cn2cccn2)NC(=O)OC(C)(C)C)=O)CCC2(COC(=O)N2)C1 C1(CC(=O)N(C2(C(N3C(C(=O)OC)CC3)=O)CCC2)C2CC2)CCCOCC1 C(=O)(C1CC(=O)c2ccccc21)NCCCNC(C(F)=C(C)C)=O c1(NC(C2C(C(=O)Nc3cc(O)cc(Cl)c3)C2)=O)ccc2oc(O)nc2c1 N1(C(COC)C)CCn2ncc(CN(C(=O)Cn3nc(C)cc3C3CC3)CC)c2C1 CC1CC(C(=O)N(C)Cc2ccsc2)N1C(=O)Cn1ccnn1 c1(C(N2CCC(NC(CC(CCC)C)=O)(CF)C2)=O)ncc([N+](=O)[O-])cc1C c1(C(N2CCC(C(C)(C)NC(CSSC)=O)CC2)=O)cnn2c(Cl)cccc12 c1(CNC(C(n2cccn2)N(C)C)=O)ccc2c(c1)CCN(C(C1(C)CC1)=O)C2 C(=O)(C1=CCS(=O)(=O)C1)NCC(CC(C)C)(C)NC(C1CCC(C)(C)O1)=O CCC(CC(=O)NCCC(=O)NCCN(C)CC)C(C)C c1(C(=O)NCC2C3(CN(C(C4N(C)C(=O)CC4)=O)C3)CC2)cnc2ncccn12 c1(OC)ccc(COC(C2(C)CCC(F)(F)C2)=O)c(F)n1 Cc1ccncc1C(N1CCC(C(F)C(=O)NCCCCN(C)C(C)C)C1)=O N1(C(c2cn(C(C)(C)C)cn2)=O)CCN(C(C23CC2C3)=O)CC1CC(F)F.CN c1(NC(C2CC(F)(F)CN2C(=O)C=CC2CC2)=O)c(Cl)cnnc1Br C(c1cccc(F)c1Cl)=CC(N1CC(NC(C(C)=CC)=O)CC1(C)C)=O C1(C(=O)NC(C(C)C)c2cncs2)CC1C1CN(C(=O)CC2CCCOC2)C1 c1(NC(C23CC(C(=O)NC(C(COCC)C)=O)(C2)C3)=O)cc(F)c(F)c(Cl)c1F C(c1cncc(C)c1)=C(C)CN(CC(=O)NC(=O)CCOc1cccnc1)C C(=O)(CCCCC(F)F)NCC1C=CC(NC(c2cc(OC)n[nH]2)=O)C1 c1(CC(=O)NC(CN(C2CC2SCc2ccccc2)C(=O)OC)=O)cnc(C)s1 c1(C(=O)NC)cc(C)nc(N2CCCC(CCNC(=O)Cc3cc(C)ns3)C2)n1 c1(NCC2CC(=C)C2)[nH]c(=NC(CCO)C2CCC2)nc2ncn(CC)c12 N1(C(C(C)Sc2ccccc2)=O)CCN(C(=O)CS(N)(=O)=O)C(C2CCC2)C1 c1(C(N(C2CC(NC(c3cc(OC)n[nH]3)=O)C2)C)=O)cccc2ncc(C)n12 Cc1cc(C(=O)N=c2ccn(C3CCOCC3)[nH]2)c(N)c(F)c1 Cc1cc(F)cc(C(N2CC3C(CNC(C4(C)CCCC4(F)F)=O)C3C2)=O)c1O N(C1CCOc2ccc(Br)cc21)C(c1c2cc(Br)ccc2nn1C)C N1(C(CCOCC#C)=O)CC2CN(C(=O)CCc3cncnc3)CC12 c1(C(N(CC(C)C#N)C2CC2)=O)c[nH]nc1CCNC(=O)C=Cc1cocn1 c1(NC(C2N(Cc3ccc(C(=O)OC)s3)CC(O)C2)=O)cc(CO)c(Cl)cc1Br c1(C(N2CCC(C3N(c4snc(C)n4)CCCC3)C2)=O)ccc(C)c(F)c1 C1(C(N(C2CCN(C(c3ccccc3)=O)C2)CC#C)=O)CC(=O)N(CC)C1 C(C)(C(C)C(=O)NCCC12CCCC1C2)NC(C1C(COC)CC1)=O CC(C)(CNS(=O)(=O)CC1CC2OCCC2O1)CCC#N c1(N2CC(NC(C(=C)Cc3ccccc3)=O)C(F)C2)ncc(Br)c(O)n1 CCCCC(C(=O)NC1CCC(NC(=O)C(N)=O)CC1)ON=C(C)C Cn1[nH]c(=NC(=O)NC2CCC(c3ccc(Br)cc3)C2)cc1N c1(OC)ccc(O)c(C(=O)N(CC(C)NC(=O)Cc2cc(C)ns2)C)c1 Cc1nnc(CC(=O)NC2(C)CC(NC(C3(F)CCOC3)=O)C2)o1 c1(N2C3(CNC(C4(Cl)CC4)=O)CC(C2)C3)ncnc2[nH]ccc12 n1(CCCOCC)cc(C2CC(NC(=O)CC3(C)OCCO3)C2)nn1 C1(C(N2CC(C)C2)=O)CC(F)CN(Cc2ccc(SC(F)(F)F)cc2)C1 c1(C(C(=O)NCCCOC)Sc2cccs2)ccc(OCCCC(C)(C)O)cc1 CCCC(C(=O)OC)C(=O)N(C1C2CN(C(c3cnn(C(C)C)c3)=O)CC12)C N1(C(c2cc(CC)cc(Br)c2)C(=O)NC(C)(C)C)CC2(CCCO2)C1C1CC1 c1(C(=O)NCC(CC=C)NC(=O)C(C)(C)C2CCCC2)cncnc1C C(=O)(CS(=O)(=O)c1ccccc1Cl)NCC1CN(C(c2c(CC)cc[nH]2)=O)C1 c1(CCC)cc(C(=O)NC(C)CC(C)NC(=O)CN2CC(C)C2)sc1C C(C(CNC(C1CCCCS1)=O)S(C)(=O)=O)NC(C1(CCCC)CCC1)=O Cc1nc(-c2cn(CC(C)NC(c3cncc(NC(N)=O)c3)=O)nn2)sc1C C(C(CC)(CC)NC(=O)COc1cccc(O)c1)NCC.N12CCCC1C2=O c1(NC(=O)OC)ccc(Cl)cc1-c1ccc(C(=O)Nc2cc(C)cnc2F)cc1 c1(C(=O)NCC(CNC(C(C#C)(C)C)=O)O)cc([N+](=O)[O-])c(C)cc1C N1(Cc2ccsc2)CC2(CCC(c3ccccc3)CC2)C1.c12nc-1co2 C12(C(=O)NCc3c(C(=O)NCc4nc(C)c(C)s4)cccc3)CCCC1CCC2 N1(C(CC(C(F)F)NC(c2c(C)ccs2)=O)=O)CCC12CCN(C)C2 C1(CNC(C(CCC)(C)O)=O)CN(c2ncccc2C(=O)NC)CCC1(F)F N1(C(c2cc(OC)ns2)=O)C(C(=O)NC2CNC(=O)OC2)CC2CCCC12 n1(CCC)nccc1C(N1CC(N(C(=O)Cc2ncc(C)s2)C)C1)=O NS(=O)(=O)c1cc(C(N2CCC3CN(C(C4CC=CC4)=O)CC3C2)=O)c(Cl)o1 C1(C)(CC)C=C(C(=O)NC2CCN(C(=O)C(C)N(C)C)C2C(C)(C)C)C1 CCC(CC)C(C)C(=O)NCC1CCCC1NC(C12CC=CCN1CCC2)=O N1(C(c2c(C)cc(C)nc2)=O)CCN(C(C2CN3CCC2CC3)=O)CC(C)C1 c1(CC(=O)NCC(CC)NC(=O)C=Cc2cn(C)nn2)oc2ccccc2c1C c1(CC(N2CCC(Cn3cc(CCN(CC)CC)nn3)C2)=O)cncc(F)c1 N1(C(c2noc(CC)c2C)=O)CCC(C)(NC(c2cc(CC)no2)=O)CC1 C1(NC(C(C)(C)OC)=O)CN(C(c2ccc(F)cc2F)=O)CC1C1CC1 c1(CC(=O)NCC(CNC(C(CC)CC)=O)C(F)(F)F)cccc2occc12 c1(OC)ncnc(C)c1C(=O)NC1CCN(C(c2csc3nccn23)=O)CC1C C1(CS(=O)(=O)NC)CC2CC(OC(N3CCC(c4cccc(OC)c4)CC3)=O)C2C1 c1(C(N2CCC(NC(C3CC4(CC(C)(C)C4)C3)=O)C2)=O)cc2c(=O)[nH]ccn2c1 c1(C(=O)NCCOCCCNC(C=CC)=O)cc(C)c(Cl)cc1Cl C1(O)(CNC(CC=C)=O)CCN(C(C2(C(N3CCCC3)=O)CC2)=O)C1.C(=O)C C(=O)(C(C)C(=O)NC1CN(C(=O)CCc2ccccc2)CC1F)OC c1(C(N2CCC(NC(=O)CCF)C(O)C2)=O)nc(Br)n2c1COCC2 CCC(CC)(CC)C(=O)NC(C)CN1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 CC1(F)COCCN(C(=O)CC2(NC(c3cscc3Cl)=O)CC2)C1 c1(OC)cccnc1CNC(=O)C(O)CNC(=O)C(O)CSC C(=O)(CCC(C(=O)N1CC(CN)CC12CCC2)C(C)C)OC c1(CC)cc(Br)ccc1NC(N1CC(NCc2cncc(Br)c2)C1)=O C1(C(=O)NC(C2CCOCC2)CC)CC(NC(c2cc(OC)cs2)=O)C(O)C1 C1(C(N(CC(O)C(C)(C)C)C)=O)CC12CCN(C(c1cc[nH]n1)=O)C2 C#CCC(CC(F)F)C(=O)NC1CN(C(=O)C(C)(C)c2ccccn2)CC12CC2 N1(C(C(CCSC)O)=O)CCOCCC1C(N1CCC(CO)C1)=O C1(N(C(CCOCC#C)=O)C)CCC(NC(=O)C(C)(C)C2CC2)CC1 c1(C(=O)NCC(C(C)C)NC(c2c(CC)noc2)=O)cnc2c(c1)CCCC2 C12(CNC(C=Cc3n(C)cnc3)=O)CCCC1CCN2C(=O)C=Cc1nccs1 C=C=CCC(=O)NCC1(F)CC(NC(=O)C(O)CC)C1 N1(C(C(COCC)C)=O)C2CC=C(C(=O)N3Cc4cccc(C)c4C3)C1CC2 S(=O)(=O)(CC(=O)NCC1(CNC(=O)CN2CCOC2=O)CCCO1)NC c1(C(N(CCC(C(C)C)NC(=O)C(=O)NC2CC2)C)=O)cncc2c[nH]nc12 Cc1c(C(N2CCC(N(C)C(C3CN4CCCC3C4)=O)C2)=O)cncc1F c1(OC)cc(C(=O)N(CCN(C)C(c2cc(C(F)F)cs2)=O)C(C)C)ccn1 N1(C(CC)C(=O)NCCCCCNC(=O)CSC2CC2)CCCCC1CO c1(C(N(CCCNC(C2C(C)CC=CC2)=O)CCO)=O)cc2ccccc2o1 C(=O)(C=CS(C)=O)NCc1ccc(CCC(=O)N(C)CC2OCCO2)cc1 N1(C(CN2C(C)CCCC2)=O)CCC(NC(C2CCN(C)C2C)=O)C(O)C1 N#CCCCC(=O)NC1C=CCCC1C(=O)NCCOC1CCC1 C(=O)(C1CCCn2nccc21)N1C(CNC(CCOCC(C)C)=O)CN(C)CC1 Cc1[nH]nc(C(=O)NCC(C2CCCN2C(c2cnnn2C)=O)(C)C)c1C(F)(F)F c1(OCC)ccc(CN2CC3CC2C3C(=O)NCc2cc(C)nn2C)cc1O c1(NC(C2CCCN(C(C(CC)(C)C)=O)C2)=O)ccc(N)cc1C(C)(C)C C1(C(=O)NC(CCNC(c2c(OC)c(Cl)ncc2)=O)C)Cc2cc(C)ccc2S1 c1(CC(=O)CN2CCC(C(=O)N(C)C)CC2)ccc(O)cc1 c1(CCCC)ccc(NC(=O)C(C)CC)c(C#N)c1.c12c(cccc1F)CNC2=O C1(C)(C(N2CC(NC(c3cccc(OC)n3)=O)C(OC)C2)=O)CCC(C)=C(C)C1 c1(C(=O)NCC2C3N(C(c4ccc(C)cn4)=O)C(CC3)C2)c[nH]c2ncccc12 C1(C(N(CC(C(=O)OC)C)C)=O)CCOCC1NC(=O)Cc1cnoc1 CCC(CCC(=O)NCc1ccc(F)cc1)NC(=O)C(C)C#N C1(C(C)C)CN(C(=O)CC2CCC3CC3C2)CCN1C(c1[nH]ccc1C1CC1)=O c1(C(=O)NCC(CC=C)NC(c2c(C)coc2C)=O)ncccc1N=[N+]=[N-] C(=O)(CC(C(F)F)n1cccn1)NCC(CC)NC(c1oc(Br)nc1C)=O C1(CCNC(c2c(C)con2)=O)CSCCN1C(=O)C(N1CCC(O)CC1)C c1(C(=O)NC2C(C)CN(C(c3cnc(S)[nH]3)=O)C2)cc2cncn2c(O)n1 N1(C(c2cncc(OC)c2)=O)CCC(CNC(=O)COC2(C)CCC2)C(C)C1 CC(CNC(C1(C(=O)OC(C)(C)C)CC1(Cl)Cl)=O)C(=O)NNC(=O)OC(C)(C)C c1(C(=O)NCC(CCCC)NC(=O)CCc2nc[nH]n2)cc2nc(=O)ccn2[nH]1 C12(NC(=O)CN(C(=O)Cc3ccnc(O)c3)CC3CC3)CCCN(CC1)C2 c1(C(COC)NC(C2CC2c2cccnc2)=O)ccc(OC(F)F)cc1 c1(N(CCOC)C(=O)NCc2nc(C)sc2C)ccc(CC2CCC2)cc1 C1(C(=O)NCC(C(=O)NCc2onc(CC)n2)N(C)C)CCC(C)(C)OC1 c1(C(=O)NCCN(C(CC(C)C2CCCO2)=O)C)ccc2c(=O)ccoc2c1 C1(C(N2CC(OCCNC(C3CCCOCC3)=O)C2)=O)CC2CCC(C1)C2(F)F C1(CNC(C2CC(=C)C2)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccc(SC)s1 c1(CCC(=O)N(CC(=O)NCC(C)C(=O)OC)CC#C)ccn(C)c1 N1(C(C(CC)NC)=O)CCC2C1CCN2C(c1cncc(C)c1)=O N1(C(C(CC(C)C)F)=O)CCC2CCCC(C1)N2C(c1cc(F)c(O)c(F)c1)=O Cc1cc(C(=O)NC(Cn2cncn2)C(=O)NCCCCN(C)CC)ccc1O N1(C(C(CC)(C)CC)=O)CCC2(CC1)CC(C)N(C(C1CC(O)CN1C(C)=O)=O)C2 C1(CC(=O)NC2(C(=O)OC)CC2C)C(NC(=O)Cc2cc(CO)[nH]n2)CC1O C1(NC(c2nc(C(C)C)oc2)=O)CN(C(=O)C(C)(C)c2ccnn2C)CC1F O=C1CCC(C(=O)NCCCCCCNC(c2ccccc2CO)=O)=NN1 N1(C(CCN(CCC)C)=O)CCC(CNC(=O)COCCCN(C)C)C(C)C1 C1(C(=O)NCC2(F)CCC(NC(c3ccc(OC)cn3)=O)C2)CC2(C1)CC2(F)F C(=O)(CC1=NNC(=O)C1)NC(c1nnc2n1CCC2)CCOCC CC(C(=O)NC1CC2(C1)CC2NC(=O)CSCC(F)(F)F)S(C)(=O)=O C(CC(C)C)(C(=O)NCC(C)(C)NC1CC1)NC(CSCCC)=O c1(-c2c(C(=O)Oc3ccc(C(=O)OC)cc3)nnn2C(C)(C)C)ccc(F)cc1C CCC(C)CC(C(=O)NC1C(C)C1C)NC(=O)CS(=O)(=O)NC C1(F)(C(N2CC(CNC(C3CCOC3)=O)C2)=O)CS(=O)(=O)CC12COC2 C1(NC(CC=CC)=O)CN(C(c2sc(C)cc2C)=O)C(CC)(CC)C1 c1(OC)c(C)cc(C(N2CCCC(NC(=O)C(C)SC(C)C)C2)=O)cc1Cl C(CCC(C)(C)CNC1(c2nnnn2C(C)C)CCCOC1C1CCCC1)OC c1(C(C)C)nc2[nH]ccc2c(=NCC(C)(C2CC2)OC)[nH]1 c12ccc(cn1)COC(=O)C2(F)F.C(CC(=O)NC(=O)OC(C)(C)C)OC C1(C(=O)NC2C(NC(c3nccc(Br)c3O)=O)COC2)CCn2nccc2C1 CCC(CN(C)C)CC(=O)N(CCCNC(C1Cc2nccn2C1)=O)C1CC1 CC1(C(=O)NC2CCC(O)C2)CCCN(C(c2ccnc(O)c2F)=O)C1 C1(CNC(CC2C(C)(C)COC2)=O)CN(C(C2(C(F)F)CC(O)C2)=O)CC1(C)C c1(COC)c(C(N2CCCCC(NC(=O)C3=CCSC3)C2)=O)oc2ccccc12 C(=O)(CCCS(C)(=O)=O)NCC1(NC(=O)Cc2ccno2)C(C)CCCC1 c1(C(N(CCCCN(C(=O)C(F)=CCCF)C)C)=O)c(C(F)F)cnn1C CC1CCN(C(c2cc(O)ncc2F)=O)CC1CC(=O)NC1(C(F)(F)F)CC1 C#CC1CN(C(C2CC(=O)CS2)=O)CCN1C(C1CC(=C2CCC2)C1)=O C1(C(=O)NCC2(C)CC(NC(c3nc(Cl)c(Cl)s3)=O)C2)CCOC1(C)C C1(N(C)C)CC(C(=O)NC2CC2CNC(=O)Cc2cncs2)C1 S(=O)(=O)(c1ccc(F)c(Cl)c1)NCCCC(=O)NC1CC1CNCc1nccs1 C1(C(=O)NC(C)(C)C)CCN(C(c2ccc(CO)o2)=O)CCO1 C1(N(C)C(c2ccoc2)=O)CC2CC1N(C(c1cn(C3CC3)cn1)=O)C2 c1(C(C(=O)N(C)CC2CN(C(c3cnc(C(C)C)s3)=O)C2)(F)F)ccccc1F CC1CN(C(=O)CCCCC2CCCC2)CC1CNC(c1cnn(C2CC2)c1)=O C1(C(C)NC(CC(=O)NCC)=O)CN(C(c2ccncc2F)=O)CCO1 CC1CN(C(=O)CCn2ccnn2)CC(C)C1NC(C1(C)C(C)(C)C1(C)C)=O C1(NC(COC2C(CC)CCCC2)=O)(CO)CCCN(c2ncc(C)c(C)n2)C1 C(=O)(C(CC)C(=O)N1CC2(C)CC1(C(=O)NC1CN(C)CCC1O)C2)OCC c1(C(C)NC(N2CCN(c3cccc(C)n3)CC2)=O)ccc2[nH]ccc2c1 C1(C(N2C(CNC(=O)C3=CCCC3)CC3(CCC3)C2)=O)CCc2ncccc2C1 c1(OC)ccc(F)c(NC(C2CC2C(c2ccccn2)Nc2ccc(C)nc2)=O)n1 CC1CN(C(C2CCCC(CF)C2)=O)CC(C)C1NC(=O)Cc1cscn1 N1(C(C2(C#C)CC2)=O)CCCN(C(C2CCC(C(N)=O)CC2)=O)C(C(C)C)C1 c1(C(N(C(C)C)CCNC(C2CC(C#N)C2)=O)=O)c(CO)nn(C)c1C1CC1 CC1CN(C(c2cscc2F)=O)CCN1C(=O)CCc1cnc(C2CCC2)o1 N(C1c2cc(C)ccc2CC1C)C(c1c(CCCCC)scn1)=O CN1CCN(C(=O)Cc2cocn2)C(C(=O)NCCCc2cc[nH]n2)C1 c1(C(N(CCC)CCNC(C2(C3CC3)CCC2)=O)=O)cc2c(C)cc(F)cc2[nH]1 c1(C(N2C(C)(C)CC(CNC(=O)CCNC(N)=O)C2)=O)ccc2c(c1)C=CCC2 N#CC1(C(F)F)CCN(c2ncc(C(=O)NC=O)o2)CC1 C1(C(N2CC(CNC(C3CC(=C)C3)=O)C3(C2)CCC3)=O)CCc2nccn2CC1 N1(C(C(CC)(C)O)=O)CC(F)(F)CC1C(N1CCC(CN=[N+]=[N-])CC1)=O N1(CCC)CCCC(C2CCOCC(C(N(c3ccccc3Br)C)=O)C2)C1 c1(C(=O)NCC2(CCNC(C(CC)O)=O)CC2)[nH]c(=N)ccc1C c1(C(=O)NC(C(C(C)C)NC(C2CC3(CC(=C)C3)C2)=O)C)cccc2ccsc12 NS(=O)(=O)c1ccc(NC(C2CNCCN2Cc2cccc(F)c2I)=O)cc1 C(C(=O)NN1C(=O)NC(c2ccccc2C(F)(F)F)C2=C1C(C)NC2=O)=CC c1(OC)cc(C(=O)NCC2(SC)CCC2)c(Nc2cc(C(C)C)ccc2Cl)cn1 c1(C(=O)NC2CC(CNC(C3C(C(C)C)(CC)C3)=O)C2)cc(F)cc(C)c1N c1(C(=O)NC2CCC(N(C(C=COCC)=O)C)C2)cc(C)nc(C)n1 N1(C(CC2C(CNC(C(C(=C)C)(C)C)=O)C2)=O)CCCN(CC)C(=O)C1 C1(NC(C2=CCN(C(C(C)(C)OC(C)=O)=O)C2)=O)CCn2ccnc2C1 C1(C)(CC(N2CCC(C(=O)NC(COC)C(C)C)C2)=O)CCOCC1 C1(COC(=O)CO)CCCN(C(=O)OCCOc2ccc(Br)s2)C1 CCCCCC(C)C(=O)N1CC(NC(c2n[nH]c3c2CCCC3)=O)CC(F)C1 c1(N(C)CC2(CO)CC2)nc(N2CCCC(C)(F)C2)nc2c1SCC2 C(=O)(C#CC1CCCC1)NCC(CC)(C)C(=O)NC(c1ncn(C)n1)C C1(C)(C(=O)NCC(CN(C)C(c2ccc(C(C)(C)C)nc2)=O)O)CCC(=O)N1 C(=O)(C1CCCc2ccnn21)N1CCC2(CCN(C(=O)C=CC(F)(F)F)C2)C1 N1(C(C2(N(C(Cc3cc(C)n(C)n3)=O)C3CC3)CCC2)=O)CC(C)C(C)C1C c1(CN(C(C(C)CN(C)C)=O)C2CN(C(C3CC(CF)C3)=O)C2)ccc(F)cc1 c1(C(=O)NC2CCCC(NC(=O)COC3CCOC3)C2)cc(Cl)cc(Cl)c1F C1(CC2C(C(=O)OC(C)(C)C)C2)(CNC(C2CC2C(F)(F)F)=O)CCC1.C1(C)CC1 c1(OC)cn2c(cc1=O)CN(c1nc(N3CCC(C)(F)C3)c3c(n1)CCS3)CC2 CCC(CC(F)F)C(=O)N1CC(C(C)NC(=O)COC2CCCC2)C1 CCC(CCC(=O)N(CCC(C)NC(c1ccc(CO)cn1)=O)C)OC C1(C)(NC(c2c(CC)cco2)=O)CCCCC1C(=O)NCCC1CCNC(=O)C1 c1(C(N2CCC(N(C(=O)Cc3cccs3)CC)C2)=O)cccc2nc(O)ccc12 CC12CN(C(C3CCO3)=O)CC1(C)CN(C(c1cccn3ccnc13)=O)C2 O=C(NNc1ccc(Br)nc1)C(=O)NC1CC(O)C12CCC2 C(=O)(C1=CC(C)(CC)C1)OCC(c1cc(C)n(CC=C)c1C)=O C1(C(=O)NCCC(=C)CNC(c2ccc(Br)s2)=O)CCC(C)(C)C1 c1(OCC(=O)NCC(C)(CO)NC(C(F)=CC)=O)ccc(OC)cc1 CC(CC(=O)NC1CCC(NC(=O)C(c2ccc(O)cc2)=O)C1)CC(F)(F)F C1(NC(C2CN(C(=O)NS(C)(=O)=O)C2)=O)CCN(C(=O)CCNCC2CC2)CC1 C1(N(C(=O)CCC2CCCOC2)C(C)C)COCCN(C(=O)C(C2CCCCC2)F)C1 c1(OCC=C)c(C(N2CCC2CNC(=O)CC2CCCC2(F)F)=O)cccc1C c1(NC(=O)CC2CCCO2)cnc(N2CCNCC2)s1 c1(CC)cccc(C(=O)NC(CNC(C2(C)CC3CC3C2)=O)C2CC2)c1O C1(C(N(C)CC2(NC(c3cccnc3S)=O)CC2)=O)CC2CCC(C1)O2 N1(C(CCC=CCC=C)=O)C2CCC1(CNC(c1cc(CC)[nH]n1)=O)CC2 Cc1cc(C(=O)NC2CC(N(C(=O)CNc3nccs3)C)C2)sc1Br c1(C(=O)NCC(CN(C(C(C)n2cccc2)=O)C)O)cnc(-c2ccccc2)[nH]1 N1(C(CSCC(C)C)=O)CCC2(CNC(c3cc(Br)n[nH]3)=O)CCCCC12 CC(C)C(C(=O)NCc1cn(C)cn1)C(C)NC(c1cccc(F)c1)=O C1(NC(C=C(CC)C)=O)CC2(CCCN(C(=O)C3=CSCCO3)C2)C1 N1(C(C(CC)(C)C)=O)Cc2ccc(C(=O)Nc3cnc(C(F)(F)F)s3)cc2C1 N1(C(C(C2CC2)NC(C=CC(=O)N(C)C)=O)=O)CC2(C=CCO2)C1 N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(=O)C(COC)N(C)C)C(CC2CC2)C1 C(CNC(=O)NC(c1ccccc1Cl)C)(CC(C)(C)C)OC Cc1cccc2c1OCC2C(=O)NC1CCN(C(=O)CC(F)(F)C(C)C)C1 N1(CC(=O)NC(c2csc(-c3ccco3)n2)C)CCc2ccc(Cl)cc2C1 N1(C(C(C)CC(N)=O)=O)CC2CCCC2(NC(c2cn(C(F)(F)CO)nn2)=O)C1 CCCC(C(=O)N1CC(C(C)(C)O)(CNC(C2CCOC2=O)=O)C1)OC c1(SC(C)(C)C)cccc2[nH]cc(C(=O)NNC(c3c[nH]c4nccc-4c3)=O)c12 C1(NCc2ccc(SC)cc2)CCCN(CC2CCNC2=O)CC1 N1(C(c2n(C(C)C)ccn2)=O)CCC2(CC2)CC1C(=O)NCC1CC1C1CCC1 c1(NC(c2cccc(Cl)c2)c2n(CC)nnn2)ccc(OCC(C)C)nc1 C(C(C)(C)CC(=O)NOCCOc1ccncc1)NC(Cc1nc(C)sc1)=O N1(C(c2cc(C)sc2)=O)CCC12CN(C(=O)CN1C(C)CCC1C)C2 C1(C)(CNC(CCC(=O)NC)=O)CN(CC2CCCC2)CCO1 N1(C(c2cccc(C)c2)=O)CCC(NC(C2C(C)C2C)=O)C(O)C1 C1(C(=O)NC(C2CC2NCCc2cn[nH]c2)C)CCC2(CC1)CC2 Cn1cc(OCC(=O)NCC2COC(CNC(c3ccccc3)=O)C2)cn1 C#Cc1c[nH]nc1C(=O)NCC(C1CC1)NC(=O)CCNC(=O)CO.C1(S)CCCC1 c1(CC(=O)N(C(CNC(C(Cc2ccc(C)cc2)C)=O)C)C)cn2ccsc2n1 c1(C(=O)NC2C=CC(CNC(COCCC#C)=O)C2)cc2cc(Cl)cnc2[nH]1 Cc1cc(C)n(Cc2cn(C3CCC(C(=O)N(CCC4CCC4)CCO)C3)nn2)n1 C1(NC(c2cnc(C)nc2O)=O)CCCC2CN(C(c3cc(Cl)no3)=O)CC12 C1(O)(C(N2C(c3cn(CCCNS(C)(=O)=O)nn3)CC2)=O)CCCCCC1 c1(C(N2CCC(C(C)(C)C)CC2)=O)cc(C(F)(F)F)cc(N)c1 CCC(C)C(=O)C(=O)NCc1ccoc1C(N1CCNC(=O)CC1)=O N1(C(CC(C)(C)OC)=O)CC(NC(=O)CSc2ccc(C)cc2C)CC2(CC2)C1 c1(OCC)cccc(C(N2CC(NC(C3CCC(F)(F)C3)=O)C(C)C2)=O)c1 C#CCC(C)(C(=O)NCC1CCOCC1)NC(=O)CC(CN(C)C)CC c1(C2C(C(=O)Nc3c(C(N4CCC(SC)CC4)=O)scc3)C2)cc(F)cc(F)c1 c1(CC)cc(C(N2CC(O)(CN(C(=O)C(C)OCCOC)C)C2)=O)ncn1 N1(C(c2cccc(CC#N)c2)=O)CCCC2(C1)CN(C(c1ccc[nH]1)=O)C2 n1(C(C)C)ccc(C(=O)N(CC(C)NC(=O)CCCN2CCCC2)C)n1 C1(NC(CC2(CC)CC2)=O)CC2CC1CC2C(=O)NCCc1nncn1CC C(=O)(C1CC(C)Cc2c[nH]nc21)NCCCN(C(=O)CCn1ccnn1)CC N1(C(CSC)=O)CCC2(CCOC2)C(CNC(C23CC=CC(C2)OC3)=O)C1 N1(C(c2ccc(=N)[nH]c2)=O)CCN(C(c2cocc2Br)=O)CC(O)C1 Cc1ccc(C)c(-n2nc(-c3cnn(CCO)c3)nc2-c2cn(C)nc2CO)c1 N1(C(CCCCC=C)=O)CCC2(NC(C3(CN(C)C)CC3)=O)CCCCCC12 Cc1cn(C(C)C)[nH]c1=NC(=O)N1CCOC(C(=O)O)C1 c1(OC)ccc(Cl)c(C(=O)NCC(C)(C2CC2)NC(=O)Cc2ccoc2)c1 c1(NCC)ccc(C(N)=O)cc1NC(c1nnnn1CC)C1(CC)CC1 c1(CNC(CC(CC)C)C(=O)O)noc2c1CC(C)(C)CC2 Cc1ccc(C(N2CCCC2c2cccnc2)C(=O)NC(C)(C)C)cc1Br.C(CO)O N1(C(c2cc(OC)ncc2)=O)CCc2c(cc(C(=O)O)nc2C)C1 C1(OC)CCC12CC(C(=O)NCCC1(NC(C3C(C)(C)C3(C)C)=O)CCCC1)C2 c1(C(C)OC(C2CC2(F)Cl)=O)cccc(Cl)c1F Cc1cc(Cl)ccc1CC(=O)NCCOCCNC(c1cnccc1C(F)F)=O C(=O)(CC(C(F)F)NC(C1CC(C)(C)CCO1)=O)NC(C(=O)OC)CC1CC1 C1(NC(c2c(OC)cccc2)=O)CC2(CCN(c3ncnn4cccc34)CC2)C1 CCC(C)(C#N)C(=O)NC1CC(F)(CNC(=O)C(C(C)C)NS(C)(=O)=O)C1 Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CCCC1CNC(=O)CC1CC1 C(=O)(C(C(C)C)NC(N)=O)NCCC1CC(C(N(CCC)CC2CCC2)=O)C1 c1(OC)cc(O)ncc1C(=O)NC(C)CCNC(c1ccc(NC(N)=O)cc1)=O C1(CNC(=O)CC2(SC3CC3CO)CC2)CN(C(c2ccc(F)cc2)=O)C(=O)O1 C1(NC(c2c(C)nn[nH]2)=O)CN(C(c2ccc(=N)[nH]c2)=O)CCC1C c1(NCc2c(C)nc(CCCC)nc2O)oc2c(OC)cccc2c1C N1(C(C(C(C)C)C#N)=O)CC2OCCN(C(c3csc(S(C)(=O)=O)c3)=O)C2C1 C(=O)(C(CC)C(C)C)N1C(C)(CCC(N2CCC(CC#C)CC2)=O)CCC1 NS(=O)(=O)CCCC(=O)NC1CC(NC(c2ccn3c2CSCC3)=O)C1 Cc1cc(CNC(c2cccc(N(C)C)n2)=O)oc1C.C12(CCC1)CC(=O)N2 c1(C(N2CCC(C(C)NC(c3cc(CC)no3)=O)CC2)=O)ccn2ncnc2c1 c1(C(=O)NC2C(CNC(C=CCCC)=O)CC2)cc(C)ccn1 C1(NC(CCCC=C)=O)CC2(C1)CC(C(=O)NC(c1noc(C)n1)CC)C2 C1(C(C)(C)CNC(=O)C=CCO)CCCCN1C(C1CC2CCC1O2)=O CC1CCN(C(c2csnn2)=O)CC1NC(=O)CC12CCC(C)(C1)OC2 C1(C(C)C)CN(C(=O)C(Br)=C(C)C)CCN1C(=O)C(C1CCOCC1)F Cc1nc(C(C)(F)F)ccc1C(=O)NC(C)CCCNC(=O)CC(O)C(C)C C1(NC(C(=O)NC(c2sccc2Br)C)=O)C(=O)NCC1(C)C CC1(C)CN(C(C2CN(C(=O)CC3CCC3)CC2(C)C)=O)CCC1O C1(CCCNC(CCSCC)=O)CCCN1C(c1cc(C(F)(F)F)c[nH]1)=O C1(C(=O)NC2CC2SC)(CC)CCCN(C(c2cncn(C)c2=O)=O)C1 N1(C(c2ncn(C)c2)=O)CCC12CN(C(=O)CNS(=O)(=O)c1cccs1)C2 C1(NC(C(CCOC)C)=O)CC(F)CN(C(c2c(Cl)c(C)nn2C)=O)C1 C(CNC(=O)COC(F)F)(CC(F)(F)F)NC(c1c(C)nc(CCCC)s1)=O C(=O)(CC1OCC(C)c2ccccc21)NC1(C=C)COC1 c1(CC)ccnc(C(N2CC(CNC(=O)CC=CC(C)(C)C)CC2C)=O)c1 N#Cc1sccc1C(N1CCC(NC(C2CCCC(C(F)(F)F)C2)=O)CC1)=O N1(C(c2cc(CC)no2)=O)CC(C)CN(C(c2c[nH]ccc2=N)=O)CC1C N1(C(c2n(CC)ncc2)=O)CC2CCC1CN2C(c1nccc2[nH]ccc12)=O Cn1cnn(CC(=O)NC2(CNC(=O)CC3C=CCC3)CC(F)(F)C2)c1=O C1(CNC(=O)CC(F)F)C2CN(C(c3cccc(-n4nccn4)c3)=O)CC12 c1(C(=O)OCC)ccc2c(c1)C(NC(C)C(=O)NC1CCC(F)(F)CC1)CCC2 C(=O)(C1CC(=O)N(C)c2ccccc21)NCCN(C(c1cnc(CC)[nH]1)=O)CC C(=O)(C#CC1CCOC1)N(C1(C(=O)NCC2OCCN(CC)C2)CC1)C C=CCCCCCC(=O)NCC(CNC(C1(C)CCCNC1=O)=O)S(C)(=O)=O N1(C(C2CC(CC)C(=O)CC2)=O)CC2CCN(C(=O)C(F)C(C)(C)O)CCC2C1 C(C(CO)CC(C)C)NC(C1(CCNC(C(C=C)O)=O)CCCC1)=O N1(C(C(CC=C)CNC(=O)Cc2cccc(F)c2)=O)CCC2(CNC(=O)N2)C1 c1(NC(=O)CC2CC(n3cncn3)C2)ccc2[nH]cc(-c3nn[nH]n3)c2c1 N=c1[nH]c(=NCC2C3COCC23)[nH]c(=NC2CC3CSCC3C2)[nH]1 N1(C(C(CC)n2nccc2C)=O)CC2=C(C1)CN(C(c1cc(C)ccc1O)=O)C2 C(=O)(C1(C)CCc2ccccc21)N1C(CN(C(CCN(CC)CC)=O)C)CCC1 C1(CNC(CC(CC)C)=O)CCC2CN(C(=O)CNC(C3CC3C)=O)CC12 N1(C(C(C(C)C)C)=O)CC(C(=O)N=c2ccn(CC(N)=O)[nH]2)C(C2CC2)C1 Cc1c(C(N2CCC(C)(CCNC(C3C4CCCCC34)=O)C2)=O)cccc1N c1(CNC(C2N(C(CCNC(C)=O)=O)CC2)=O)cccc(C#N)c1 CCC(C)(CO)C(=O)N1CC(NC(c2occc2CSc2ccccc2)=O)C(C)C1 CCC(c1ccc(C)cc1)=CC(=O)NCC(C)NC(=O)C(C)(C)CC(C)C C1(CNC(C=NOC)=O)N(C(=O)Cc2ccc(C3CCC3)cc2)CCCC1(C)C c1(C(N2C(CCNC(C(C)SC)=O)CCC2)=O)ccc(C2CNC(=O)C2)cc1 c1(CNC2C(COC)CCCC2)cccc(OC)c1F c1(C(=O)OC2CCCC2NCC(O)C(F)F)ccc(O)cc1F C(=O)(CC(C)CC(=O)NCC1(C)CCCN(C(=O)CCNC(=O)CO)C1C)OC Cc1ccc2c(c1)CC(C(=O)NC1CC(C)(NC(=O)C(n3nccc3C)C)C1)S2 N#Cc1ccc(CN2C(C(=O)Nc3cncc(C4CC4)c3)CC3CC23)c(Br)c1 N#Cc1ccc(F)c(-c2ccc(CO)o2)c1Cl c1(C(=O)NC(CCOC)CNC(c2cnn(C3CC3(F)F)c2)=O)n[nH]c(C)c1O N1(C(c2nc(C)n(C)c2)=O)CCN(C(=O)CC2CC23CC3)C(c2ccccn2)C1 C1(C(=O)NCCCCCCC)CN(C(c2cnc(C)s2)=O)CCC1(C)C c1(NC(=O)CC2CCN(C(=O)CN3CCCCCC3)CC2)cc(O)cc(F)c1 CP1(=O)CCN(CC(=O)NCCNc2ccc(-n3ccnc3)cc2)CC1 c1(C(C)(F)F)ccnc(NCC2(O)CC(CO)C2)n1 Cc1ccc(C=CC(=O)NC2CCC(N(C)C(c3sccc3C#N)=O)C2)cc1C C#CC1C(C(=O)NC(C)CN(C)C(c2ccnc(OCC(F)F)c2)=O)C1(C)C c1(C(=O)NCC(C)N(C(C(CCCOC)C)=O)C)cc2c(cn1)CCCC2 C1(C(N2CCC(C(=O)NCC3(C)CCCCO3)CC2)=O)CC2(CCC2O)C1 N1(C(c2ccc(C)nc2)=O)CCC2CN(C(=O)C=CC3CCCCCC3)C2C1 CCCC(C(=O)NCC1(C)CCN(C(=O)CCc2ccccc2Cl)C1)NC(N)=O CCC1=C(C(=O)NC2CCN(C(C3(C)CCC(=O)C3)=O)CC2(C)C)CCCO1 Cc1ccn(C)c(=O)c1NC(C1CN(C(=O)Cn2c(O)nnc2O)C(C)(C)C1)=O c1(NCC2(NC(=O)CCC3CCCCO3)CCCC2)ncc(O)cn1 N1(C(c2ccn(CC#N)n2)=O)CC2CN(C(C3CSCCS3)=O)CC2C1 C1(C)(C(CC)NCC)CCC2(CC1)OCCO2.CC1(C#CC(=O)N2CCC2C)CC1 CC#CCCC(=O)N1CC2C(CNC(=O)Cc3sc(S)nc3C)C2C1 C1(C2(O)CCN(C)CC2)(OCCOC(c2nn3cccc(C)c3c2)=O)CC1 N1(C(C2CC(CC)C2)=O)CC2CCC1CC2NC(=O)Cc1cc(C)on1 C(=O)(CC(F)(F)C(F)F)NC1C(NC(=O)Cc2cc(Br)ccc2O)CC1 c1(OC)ccc2c(c1)C1(CC1)CN(C(c1cc3cc(Br)cn3c(Cl)n1)=O)C2 C(=O)(CC(F)(F)C(=O)O)N1C2CN(C(=O)C=CC3CC3)CC21 CCCC(C)(O)C(=O)N1CCC(F)C(NC(=O)CCc2nc(C3CC3)no2)C1 C(=O)(CCC(=O)NC(C(=O)NC(C1CCCC1)CO)C1CCCO1)N(C)C n1(CC(C)NS(c2c(C(=O)OC)scc2)(=O)=O)cnc2c1c(=O)n(C)c(=O)n2C c1(OCC)cc(C(=O)OC)ccc1NC(=O)COC(c1cnn(C2CCC2)c1C)=O n1(CC)nnc2cc(C(N3CCC(NC(=O)CCS(C)=O)C34CCC4)=O)ccc12 C(=O)(C(CC)(CC)CC)NCCC1CCN(C(c2cccc(CC)c2F)=O)C1 C1(C(N(C)CC2CN(C(c3ccn(C(F)F)n3)=O)CCO2)=O)CCCCCN1C CC(C)C(O)C(=O)NC(CC1CC1)CC(=O)N1CCC(OC2CCC2)C1 C1(CN(C)C(c2cc(Br)n(C)n2)=O)CN(C(C2CCCCO2)=O)CC12CC2 Cc1cc(-n2cc(-c3n(CCO)nc(C4CC4)c3)nn2)cc(Br)c1 C#CCCCCC(=O)N1CC2(CC(CNC(=O)C(C3CCCCC3)O)C2)C1 Nc1ncc(Br)cc1C(N1CC(NC(=O)CCc2cnn[nH]2)C(O)C1)=O N1(C(COCCC(C)C)=O)CSCC1C(=O)NC(C1CCN1C)C1CC1 N1(C(C)=O)CSCC1C(=O)NC1CC(CNC(C2CCC2)=O)C1 N1(C(CC2N(C(Cn3c(C)nc(C)n3)=O)CC2)=O)CCCC(C)C1CO c1(CNC(C(=O)NCC)=O)cccc(C(N2CCC(CO)C2)=O)c1 CCCCCCC(C)C(=O)N(CC(C)N(C(=O)C(COC)N(C)C)C)C c1(N2C(C)(CNC(COc3cccc(C)c3)=O)CCC2)ncc([N+](=O)[O-])cc1Cl N#CC1(C(=O)Nc2cccc(CNC(=O)C(=O)NC3CC3)c2)CC2CCC1C2 N1(C(CCN2CCN(C)CC2)=O)CCC=C(C(=O)Nc2cnc(O)nc2O)C1 c1(NC(N2C(C3(NC(C4C=CC=CC=C4)=O)CC3)CCC2)=O)ccccc1F C(=O)(CS(=O)(=O)c1ccccc1F)N1CCN(C(C2C(C3C(C)C3)C2)=O)CC1 N1(C(c2ccc(CC=C)cc2)=O)CCC(C(=O)OC)CC1CC Cc1ccc(C(=O)NCC2CC(F)(CNC(=O)Cc3nc(=N)[nH][nH]3)C2)nn1 c1(C(=O)NCC2(NC(c3nc(C)sc3)=O)CC2)ccc(Br)c(C(F)(F)F)c1 C12(NC(C(C)N(C)C)=O)CC(C)(C1)OC21CN(C(C2CC3(CCC3)CO2)=O)C1 C1(C(=O)NCCC2CCCN(C(C(CO)OC)=O)C2)CCCCCN1C N1(C(C(C)OC)=O)CCC(C)C(NC(=O)C(N2C(=O)CCC2=O)CC)C1 C(=O)(CCCCCNC(=O)C(C1CCCCC1)=O)NCCc1n(C)cnn1 CC1(NC(=O)CN(C23CCC2CC3)C)CN(C(=O)COc2ccccc2)C1 CC1C(NC(=O)CC23CCC(CC2)C3)CCN1C(c1c[nH]c(C(F)(F)F)c1)=O c1(CN(CCC(=O)N(CCC)CCC)CCOC)ccc(Cl)c(O)c1 O(NC(=O)CC(C)NC(c1c(C)cnnc1O)=O)C(C=C)C N1(C(COC(CC)(C)C)=O)CCN(C(c2nscc2C)=O)CC(O)C1 c1ccc2c(=NCCCn3ccnc3)[nH]c(NC3CN4CCCC3C4)nc2c1 N1(C(CCSC)=O)CCCC1CCC(=O)NC(CO)C(N)=O N1(C(Cc2c(C)cccn2)=O)CCOC2CN(C(=O)CCc3ccsc3)CC12 C12(C(=O)OCC)CCCC1CN(C(c1ccc(C)c(I)c1)C(=O)NCCC#N)C2 C(=O)(C1(C)CCn2c(C)nnc21)N1CCC2(CCN(C(C3CC(=C)C3)=O)C2)C1 CC(C)C(C)C(=O)N1CC(C(O)C(=O)NC2CC(N3CCCC3)C2)C1 c1(C(=O)NCC(C)(C)NC(CCc2c(C)ncnc2O)=O)cc2n(n1)CCOC2 C1(CNC(c2ccc(C(F)F)c(F)c2)=O)CC2CCC1N2C(=O)CSC(F)(F)F C1(OC)CN(C(=O)CCc2cnc[nH]2)CC1NC(c1sccc1OC(F)F)=O N1(C(c2c(C)nc(CCC)s2)=O)CCN(C(C2CSCCS2)=O)C2CC12 C1(CC(C)NC(=O)CC2(O)CCCC2)CCN(C(C2CCCCCC2)=O)CC1 C1(OCCC)CCCN(C(C2CCC(NC(=O)Cc3nonc3C)CC2)=O)C1 C1(C(=O)NCCC2(O)CN(C(c3c(C)cc(O)nn3)=O)C2)CN(C)CCN(C)C1 C(=O)(C(C)CCNC(=O)C(CC1CC1)NC(C12CCC(C1)C2)=O)OC n1(CC(N2C(C)CC(NC(c3ccc(SC)o3)=O)C2)=O)ncn2cccc2c1=O c1(OC)cc(F)c(S(N)(=O)=O)cc1C(=O)NCCNC(=O)CC1=CCCC1 CC1(C)CC(S(N)(=O)=O)CN1Cc1cc(CO)cc(Br)c1 N1(C(C2(C(=O)NCc3c(SCC)[nH]cc3)CC2)=O)CCC2(CC1)CC(CNC)C2 CC1OC2(CNC(=O)CC3NC(=O)NC3=O)CC1(NC(c1cnccn1)=O)C2 C1(NC(C2COCCO2)=O)CCN(C(c2ccc(-c3ccccn3)o2)=O)C12CC2 C1(C(=O)NCC2(NC(C=C(CC)C)=O)CCC2)CCCN1C(=O)C(F)(F)F Cn1ccc2[nH]c(C(=O)NCC3CCCC3NC(c3coc(CO)c3)=O)cc12 c1(CC)ccc(NC(C(C2(C)CC2)NC(N2CCC(OC)C2)=O)=O)cc1 N1(C(CCNC(COC)=O)=O)CC(C)(C)CC1CNC(c1cn(C)cc1C)=O c1(C(=O)NCC2(C)N(C(C=C(C)C)=O)CCC2)cn(C)c(=O)c2cncn12 N1(C(CC=CC=C)=O)CC2CC2(CNC(C2CSCN2C(C2CCC2)=O)=O)C1 c1(C(C(=O)NC(C)C(=O)OC)N(CC=C)CCC)cccc(Cl)c1.C(C1CC1)N n1(CC(=O)NCC2CN(C(C3CC4C=CC3CCC4)=O)C2)ncc2cccnc12 C1(NC(C(CC)n2cccn2)=O)CCCC(CC(=O)N(C2CCC2)CCO)C1 Cc1cc(NC2CC(C)N(C(c3cc(C4CCC4)on3)=O)C2)n2ncnc2n1 c1(CCN(S(C2CN(C(=O)C3CC3)C2)(=O)=O)C2CCCC2)cccc2[nH]ccc12 CC1C(C(=O)N2CCC(F)CC2C(N2CC(C)C(F)C2)=O)=NOC1C N1(C(CCC#C)=O)CC2(COC(CNC(=O)C(C)CN3CCOCC3)C2)C1 CCC(C)(CNC(c1nccnc1C)=O)C(=O)NCCOCC(=O)NC N1(C(CC=CCNC(=O)CCCC2CCCO2)=O)CC2CCC1CC2 N1(C(c2ccc(CNC(c3c(C)nsc3)=O)cc2)=O)CC(CN(C)C)CCC1C c1(CSC)ccc(C(=O)NC2CCC(CNC(C3CCCSS3)=O)C2)o1 Cc1c(NC(=O)N(C(C)C)C(C)C)cccc1N1CCCC1 c1(C(NOCC)=O)cnc(CNC(c2cnn[nH]2)=O)nc1 N1(C(CN(C2CCS(=O)(=O)C2)C)=O)CCC(F)(CNC(=O)C2=C(Cl)CC2)C1 C#CCCC(O)C(=O)N1CCN(C(=O)C2=CCCCO2)CC1CCO CC(CCC(C)(C)C)C(=O)N1CC2(C(=O)NC(C(O)CO)C3CC3)CCC1CC2 C(=O)(C(C)S(C)(=O)=O)NC(C(C)C)(C)CNC(c1coc(Cn2cccn2)c1)=O C1(CN(C(C2CCC(=O)N2)=O)CC)CCN(C(=O)COC(C)=O)CC1 C1(C(=O)NCC(C)CNC(=O)CC2(C)CCCCC2)COCC(C)(C)O1 c1(C(=O)NCC2N(C(CCCN(C(C)C)C)=O)CCC2C)cn2c(n1)COCC2 C1(F)(CNC(c2cn(CCC)nn2)=O)CCC(CNC(c2cocn2)=O)C1 N1(C(C(COC)C)=O)CCN(C(=O)CN(C)C)CCC1C N1(C(c2ccn(CCNC(C3(Cl)C(C(C)=O)C3)=O)c2)=O)CC2OC(=O)N(C)C2C1 C=CCC(C(=O)N(C)Cc1ccnn1C)NC(=O)COC1CC=CC1 C(CNC(C12CSCC1C2)=O)(CC(F)(F)F)NC(C1C2COCC12)=O n1(C(CC)C)ccc(=NC(=O)C(C2CCCO2)NC(=O)COC(C)C)[nH]1 c1(CNC(c2cnc(C(C)(C)C)[nH]2)=O)ccc(CNC(=O)CSC(F)F)cc1F O=S(=O)(c1cccc(=NC2Cc3cc(Br)ccc3C2)[nH]1)NCC1COCCO1 N(C(=NCCc1ccoc1)NCCCC(C)(C)C)CC(=O)N(C)C c1(C(=O)N(C2(C(=O)NCC(O)CC3CC3)CCC2)C2CC2)occ2c1CCC2 c1(C(N2C(CC(=O)NCCC(=O)OC)CCC2)=O)c[nH]nc1[N+](=O)[O-] N1(C(c2ccccc2-c2ncc[nH]2)=O)CC2CC(NC(C34CC3C4)=O)CC1C2 N1(C(C2(C)CCCOC2)=O)CC23CCCC2(C1)CN(C(C1(C)COC(=O)C1)=O)C3 Cc1ccc(CN2CCC(C)(C(N3CC4CC(C3)O4)=O)C2)n1C C1(NC(C(C(C)OC)N(C)C)=O)CN(C(c2cc(C)cs2)=O)CC1(C)C C1(NC(c2cc(C)sc2C)=O)C(C)CN(C(c2ccnc(C3CC3)c2)=O)CC1C N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(c2cc(CO)c(C)o2)=O)C2CC2C1 C1(C(=O)NCc2cc(C)cs2)(COC)CCCN1C(C)=O c1(C(=O)NC)cc(=NCc2ccccc2Cl)cc[nH]1 c1(OC)cccc(C(=O)NCCC2CCC(NC(c3csnc3OC)=O)C2)n1 O(S(=O)(=O)C1CC12CCCCC2)CCS(C)(=O)=O N1(C(C(CC)(C)C)=O)CCCCC(N(C(=O)CCCC(=O)C2CC2)C)C1 N1(C(CC(C)O)=O)CCC(O)C2(CCN(C(c3nccnc3C(N)=O)=O)CC2)C1 N1(C(C(c2cccc(C)c2)C)=O)CCCC(F)(CNC(C2CCCC3CC23)=O)C1 C1(C(N(CC(C)(C)O)CC(C)(C)O)=O)CCN(c2ccnc(Br)n2)CC1 N1(C(C(CC(C)C)ONC(C23CCCC2C3)=O)=O)CCC12CCCSC2 c1(C(=O)NCCNC(C2CC(Cl)(Cl)C2)=O)cc2ccncc2s1 NS(=O)(=O)CC(=O)NC1CCC(NC(=O)COc2ccccc2-c2cnc[nH]2)C1 C#CC1CC2(CC2)CN1C(C1(CNC(C2CCN(C)CC2)=O)CCCCC1)=O C(=O)(C(O)C(CCC)NC(c1c(C)nn(CC)c1C)=O)NC(CCC)CCC N1(C(C=C(C)c2ccsc2)=O)CC(C)CCC1CNC(c1ccc(CO)o1)=O C1(NC(c2cnc3n2CCC3)=O)CC2CN(C(=O)CN3C(=O)CNC3=O)CC12 N1(C(COCCN(C)C)=O)CCCC(C(=O)N(C2CC(C)(C)C2)C)CC1 CCCS(=O)(=O)CC(=O)N1CCSCC1CCNC(=O)C(N1CCOCC1)C C1(C(=O)NC(C=C)C2CCC2)CCN(C(=O)CC2CC(=O)C2)CCO1 CCCCC#CC(C)(C)NC(C1C=CCN1C(c1cc(CC2CC2)on1)=O)=O C1(C(=O)OC)CC(O)CN1C(C1CCC(NC(c2ccc(Br)cn2)=O)C1)=O c1(C(=O)NCC=CCNC(C2(C=C)CCC2)=O)sc(NC2CC2)nc1C CC1CN(C(=O)CC2(N3CCOCC3)CC2)CC1CNCC(C1CC(F)(F)C1)=O c1(C(N2CC3CN(C(c4cncc(C)n4)=O)CC32)=O)cccc(C)c1[N+](=O)[O-] C(C(CC(F)(F)F)OC(C)(C)C)NC12CC(C(C)(C)C)(OC1)C2 c1(C(=O)NC2C(NC(C3N(CC)C(=O)CC3)=O)CCCC2)cc(Cl)cc(Cl)c1 C1(C(=O)NCc2cc(C3CC3)no2)CN(C(c2cn(C3CC3)nn2)=O)CC1(F)F c1(-n2c(C)nnn2)ccc(C(=O)NC(C)(CNC(c2cscn2)=O)CO)cc1 c1(CCNC(=O)NN2CCC(C(C3CC3)C3CC3)C2)nc(-c2ccccc2)cs1 C1(CNC(CC2(C(=C)F)CCC2)=O)CC2(CCC2)CN1C(=O)C(C(C)C)NC=O CC(C)C(C)CN=c1[nH]c2ccc(S(=O)(=O)NCCOCCC(C)C)cc2s1 CCC(C)(C(=O)N(CCCNC(c1cnn(C2CC2(F)F)c1)=O)C1CC1)OC Cc1cc(C#N)ccc1NC(C1CCN(C(=O)COCC(C)C)C(C)C1)=O c1(CNCC(c2ccncc2)C)ccc(N)c(F)n1 N1(C(c2c(C)noc2C)=O)C2CCC1CC(CNC(C1(C)CC1F)=O)C2 CC(CNC(=O)CSCCC#N)C(=O)NC(c1ncccn1)C N1(C(C(CC=C)C)=O)CC2(CC2)CC1CNC(=O)C(C)Cc1ccco1 C1(Nc2cccc(NC(=O)NCCC)c2)CN(C(=O)CC)CC2(CC2)C1 c1(-c2n(C)ncc2NC(=O)CC2COC3CC2C3)ccc(F)cc1F c1(C(C)NC(c2cccc(OC)n2)=O)ccc(F)cc1F.C123CC1CN(C2)C3 c12cncc(c1)C(=O)N2.CC(F)(F)C(=O)N1CC(NS(C)(=O)=O)C1 C1(C2CC2)(CNC(CN(C)C2CC2)=O)CCN(C(C2CCN(CCF)CC2)=O)C1 C(=O)(CC(C)CF)OCCSc1ocnc1C(=O)NC1CN(C(=O)NC)C1 C(=O)(CCCCCN=[N+]=[N-])N1C(C)CC(NC(=O)CCOC2CCCCC2)CC1 C(=O)(CC(C)C(=O)N1CCCN(CCNC(=O)C(C)CC(N)=O)CC1)OCC CC1CN(C(=O)CN2CC(=O)NC2=O)CCCN1C(c1cccc2nsnc12)=O C1(C(N(CCCN(C(c2ccc(COCCOC)o2)=O)C)C)=O)COCCOC1 c1(OC)ccccc1C(C)=CC(=O)NC1(CN(C(=O)CC2OCCC2C)C)CC1 C1(C(=O)NCC2(OC)CN(C(C(CC)C(=O)OC)=O)C2)Cc2cc(C)ccc2S1 c1(CC(N2C(C(=O)NC(C(n3ncc(C)c3)C)C)CCC2)=O)cnn(C)c1C Cc1c(O)cccc1NC(=O)C(C)(CC)c1ccccn1 C(=O)(C(C)(C)CN(C)C)NC(C)C(CO)NC(c1nc(C(F)(F)F)cn1C)=O N1CC=C(CC(=O)N(C)C)CC1.C(C)(C)(CCCC=O)OC.C(=O)(CO)N C1(C(N2CC3CN(C(c4c(CC)nccc4)=O)CC32)=O)CCCC2CCCCC12 c1(C(N2CC(CC=C)(NC(c3csc(C)c3)=O)C2)=O)ccc(C)c(Br)c1 CP(C)(=O)CC(=O)NC1CCC(F)(CNC(c2cc(C(N)=O)co2)=O)C1 Cn1cnc(N2CCC(NC3CC(C(=O)OC(C)(C)C)=NO3)CC2)cc1=O c1(CN(CC(C)OC)C)ccc(CNC(=O)C(C)Cc2cnc[nH]2)cc1 C(=O)(C(CCOCCO)NC(C1CC(C)(C)C1)=O)NCC#CC C=CCC(CC)C(=O)NCC(C12CCC(CC1)C2)NC(=O)C(CN(C)C)C(C)C C1(CNC(c2nc(CC(C)C)sc2)=O)C2CN(C(c3cnn(C)c3)=O)CC12 CN=c1ccc(C(=O)NC2COCC2CNC(=O)Cc2ccc(SC)cc2)c[nH]1 Cc1ccc(S(C)(=O)=O)cc1C(=O)NC(c1ccnc(OC(F)F)c1)C c1(CCC(=O)NCC2CCCN(C(c3n(C)c(O)nc3)=O)C2)ccc(Cl)c(Cl)c1 Cc1n[nH]c(C)c1C(=O)NCC(Cc1ccccc1)N(C(=O)C1=CCCC1)C C=CCCC(C)(C)C(=O)N1CC2(CC)CC1(CNC(=O)Cn1cnnc1O)C2 Cn1ccc(C(N2CCC(CCNC(=O)C(C)(F)CC3CCCC3)C2)=O)cc1=O Cc1ccc(N2CC(C(=O)OCc3ncnn3C3CC3)CC2=O)c(C)c1 c1(CC(=O)N(CC(C)(C)NC(C(C(C)SC)O)=O)C)ccc(Cl)cc1F c1(CN2C(C(=O)NCC(c3ccccc3)CC)CCCC2)ccc(OC)c(OC)c1 CCC(CCCC(=O)N1CCSCC(C)C1)NC(=O)CSCC(F)F N1(C(Cc2cccc(C)n2)=O)Cc2occ(C(=O)NCC3CC(=O)N(C)C3)c2C1 CC(C)CCCC(=O)NC1C=CC(C(=O)N(CCC(C)C)C)C1 C(=O)(CCCC1N=N1)N(C(C)C(=O)N(CCO)C)CCC.C1(C)CCCO1 c1(OC)ccc(C(=O)NC23CC(CNC(=O)CCN4CCCCC4)(C2)C3)c(F)c1 C1(C(N2CC(C3(NC(C4CCCC(C)C4)=O)CC3)C2)=O)CN2CCN1CC2C CC(C)(CN(C(=O)C(C1CN(C(=O)CC2CCC(=O)C2)C1)OC)CCO)CO c1(C(=O)NC(C)C(CO)NC(=O)C(O)C(F)F)cc2c(nc1N)CCC2 C(CN=c1nc(NCCC(=O)NCC)cc(C)[nH]1)(C(C)(C)C)N(C(CCC)C)C C1(C(=O)NC(C(=O)NC2CCN(CCC)CC2)CC)CCCC2(CC2)C1 N1(C(C2(C(C)=O)CCC2)=O)CC2(C(=O)NCCCC3CC3C)CCC1CC2 c1(CN(C)C)cccc(C(=O)N(CCCNC(c2c(Cl)csc2Cl)=O)C)c1 CC(CNC(c1ccc(O)c(F)c1)=O)C(F)C(=O)NOCC1CCCC1 CCCCCCC(=O)N(C1CN(C(c2cccc(OC)n2)=O)C1)C C1(NC(COCCOC)=O)CCN(C(=O)Cc2nncn2C)CC1C(N)=O C12(C(=O)NCCCOCCN(C(=O)C=CCOC(C)(C)C)C)CC1COC2(C)C N1(C(C(CC(N)=O)O)=O)CCOC2(CCCN(C(c3ccc(C(N)=O)o3)=O)C2)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CC3CC2CN3c2ncc(C)c(C)n2)=O)n1 C1(C(C)C)CN(C(=O)CSc2nccn2C)CCCN1C(C1CCC2(CC2)C1)=O c1(C(=O)NCC2C(NC(c3cc(CC)[nH]n3)=O)CCC2)ccc2c(c1)NCCC2 C(C(C)(C)CC(=O)NC(CO)C(C)O)NC(c1cc(C(C)C)no1)=O CCCCCCC(=O)NCC1(CNC(c2ccc(CN(C)C)[nH]2)=O)CC12CCC2 c1(OC)c(C)cc(C(=O)NCC2CN(C(=O)CC3CN(C)C3)CCO2)cc1Cl c1(N2CCC(C3(C)CC3)CC2)nc2ccsc2c(=NCC2CN(C3CC3)C2)[nH]1 C(C(O)CCNC(C1CCCN1C(c1cc(Cl)n[nH]1)=O)=O)OC O=S(=O)(c1c(Br)cc(F)cc1Br)N1CCN(c2nc[nH]n2)CC1 c1(C(=O)NC(C2CC2C(N2CCC(C#N)C2)=O)C)ccc([N+](=O)[O-])s1 C1(NC(c2ccc(-c3ccccn3)nn2)=O)CCOC(CO)C1 C1(C(=O)NC2C3CC2CN(C(=O)CCC2CCCOC2)C3)CCN2CCCC2C1 CC(C)CC(C)CC(=O)NCCN1CCN(C(c2cccc3c2CCO3)=O)CC1 n1(CCCOC)ccc(=NC(=O)C2CSCN2C(C2CC(C)=NO2)=O)[nH]1 c1(C(N2CCC(N(C(C(CCC)O)=O)C)C2)=O)cccc2c1OCC(=O)N2 c1(NC(C)=O)ccc(Cl)c(C(=O)NCC2(C(=O)O)CC2)c1 c1(CCNC(c2ccc([N+](=O)[O-])cc2)C)ccc2cc[nH]c2c1 C(c1cnn(C)c1)=CC(=O)NCCCC.N1CCOC(CC(N)=O)C1 C=CCCCC(C(=O)OC)NC(=O)C(CN(C)C)NC(C1CCCCNC1=O)=O C1(NC(C2(CC)CC2)=O)CCCC1CNC(C1CC12CCC2)=O N1(Cc2onc(C)n2)CCC(NC(=O)CC(=O)N2CCOCC2)CC1C C(C(C(=O)N(CC(=O)OC1CC1)C)n1cc(-c2cnccn2)nn1)OCC Cc1cc(C(N2CCN(C(=O)CC3CC3)C(C3CCC3)C2)=O)c(Br)c(C)c1 N1(c2n(CCc3c(C)nn[nH]3)nnn2)CCC(F)(c2ccc(F)cc2)C1 N1(C(C2CC(NC(C=CC(=O)OC(C)(C)C)=O)C(O)C2)=O)CCC2CCCC2CC1 C1(NC(C2CCC(C)(C)N2C(=O)C2CC2)=O)CC2(CNC(=O)O2)C1 N#Cc1cc(Cl)c(Cl)cc1NC(C1CCCN1C(=O)CCNS(C)(=O)=O)=O c1(C(N2CCC(CC(C)NC(C3CC4CC4C3)=O)CC2)=O)ncnc2cc[nH]c12 N1(C(C2CCC(C(N)=O)O2)=O)CC(NC(C2(C(c3ccco3)=O)CCC2)=O)C(C)C1 C=CC1CC(NC(=O)C(COC)NC(=O)CCOC(C)C)CCO1 C1(CNC(C(C)NC(=O)NC)=O)CCc2cnnn2C1 c1(CC(=O)NCC(c2ccncc2)N2CCOCC2)ccc(Br)c(Cl)c1 O=C1CSCC(C(=O)NCC2(F)CN(C(C3CC(N4CC(O)C4)C3)=O)C2)N1 C1(NC(c2cccc(CC)n2)=O)CC(C)CN(C(=O)Cn2ncc(Cl)c2C)C1 N1(C(C(N2CCCC(O)C2)C)=O)CC(NC(=O)C=CC2CCC2)C(F)C1 N1(CC(C)C)CCCCC1C(=O)NCC(C)NC(=O)C=CC(C)(C)C c1(SCC(N2CC(C)C(CNC(=O)C(F)n3cccn3)C2)=O)cccc(C#N)c1 c1(C(C(=O)NCCN(C(c2ocnc2C)=O)CC)C2CCCC2)ccn(C)c1 C1(NC(=O)CCc2cnccn2)CN(C(=O)C(F)OC(F)(F)F)CCC12CCC2 CC#CCCCC(=O)NC1CCN(C(c2c[nH]c(=N)nc2C)=O)C1 Cc1cc(NC(=O)NCCc2noc(C(F)F)n2)c(Cl)cc1[N+](=O)[O-] C1(NC(N)=O)CC2CC1CN(C(C1(CNC(c3ccc(COC)o3)=O)CC1)=O)C2 C1(CNC2(c3nnnn3C3(C)CC3)C(CCCC)CC2)CCN(CC)CC1 c1(OC)ccc2c(c1)CC(C(=O)NCCCCNC(c1csc(Cl)n1)=O)CC2 Cc1cnn(CCCNC(c2nnnn2C2CCOC2)CC2CC=CC2)c1 c1(C(=O)Nc2nnc(CS(C)(=O)=O)s2)cc(OCC(F)(F)F)ccc1O c1(OC)ccc(N)c(C(=O)NCC(C)CNC(=O)Cc2nc[nH]n2)c1 c1(C(=O)NC(C)CC(C)NC(C2(O)CCOC2)=O)cc(F)c(F)c(F)c1 c1(CNC(C(C)CO)=O)cncc(C(=O)N(CC(O)CO)C(C)C)c1 CC(C)C1=NOC(C(=O)NC2(C)CCC(NC(=O)C(=O)NC3CC3)CC2)C1 c1(CNC2C(C)(C)C2)nc(Cc2ccccc2)cs1 C(CCC(C)C(=O)NC1CC2C(NC(=O)C(C)Cc3ccnn3C)C2C1)OC C(=O)(C1=CC2(CCN(C(=O)CCCn3ccnc3)C2)C1)NCC1(S(C)=O)CC1 S(=O)(=O)(C1=C2CCN=C2N=N1)NCC1C(CC)CCN1C(c1nc(CC)cs1)=O N1(C(c2ccc(C)n2C)=O)CCCC(C)(CNC(=O)C(C)N2CCC2)C1 C(C(C)(CC)N(C1CC1C(F)(F)F)C(=O)OC(C)(C)C)N.CN(CCC1CC1)C=O Cc1ncc(C(=O)NC(CNC(c2cnn(C)c2)=O)C2CC2)n1C c1(NCC2(COCC)CCOC2)ccc(S(=O)(=O)Nc2ccccc2)c(Cl)c1 C1(NC(C(c2ccccc2F)C)=O)CCOCC1NC(=O)C=CCN(C)CCO C(=O)(C(C)(C)CC(C)C)NCC(C)OCCNC(C(CC)(C)OC)=O C=CC1(C(=O)N(CCCCCC(=O)Nc2cccnc2)C)CCCCC1 C1(NC(C(c2cccc(C)c2)(F)F)=O)CCCC(=O)CC1.C12CC1CNC2=O Cc1ccc2ncccc2c1NC(C1CC(NC(=O)C#CC(C)C)C1)=O C(=O)(CCCCCOC)N(CC(CC)NC(c1nc(C2CC2)cs1)=O)CC c1(C(N2CCCC(N(C(=O)CC34CCCC3C4)C)C2)=O)cc2nc(F)ccc2o1 C1(CNC(c2cc(SC3CC3)n[nH]2)=O)CCN(c2cc(O)ncn2)CC1 c1(C(=O)NC(C(=O)NCc2cnsc2)C2CCCC2)cc2n(n1)CCO2 C1(NC(C(CCSC)OC)=O)CN(C(c2nc[nH]c2C(F)(F)F)=O)CCC1F C1(C(=O)NC(C(C)SC)C)(CNC(c2cccc(CO)n2)=O)CC(C)(C)C1 N1(C(c2cc(C)on2)=O)CC2(CCC(NCc3coc(C)n3)C2)C1 C1(N(C(c2c(CC)ocn2)=O)C)CN(C(=O)CCc2nncs2)CC12CC2 c1(CN=C(N(C)CC2CCC(CC)O2)NC2CC2)cccc2c1OCC2 N1(C(CCNC(=O)OC(C)(C)C)=O)CCC2(NC(c3ccccc3)=O)CC2C1 CC1(C(=O)NC(c2cn(-c3c[nH]ccc3=N)nn2)(C)C)CC2CC2C1 CON(C)CCCNC(=O)C(CNC(=O)C(F)OC(F)(F)F)N(C)C C1(C(NOCC(=O)NCCCC2(O)CCC2)=O)CC2(CCC2O)C1 N1(C(=O)OC(C)(C)C)CCC(F)(F)C1Cn1cc(NC(=O)OC(C)(C)C)cn1 C(=O)(C(F)(F)C1CCCC1)NCC1CC(NC(C(N(C)C)C2CC2)=O)C1 C(=O)(N=S1(=O)CCCC2(C1)OCCO2)C12CC(C(F)(F)F)(C1)C2.CCO Cc1cccc(C(N2CCC(NC(=O)CS(=O)(=O)N3CCOCC3)C2C)=O)c1C c1(NC(N2CC(C(CC)CC)C2)=O)cc(Br)cc(F)c1O C1(CNC(C(C)C2CCCO2)=O)CCN(C(C2(C)CC(C(=O)OC)C2)=O)CC1 C1(NC(C2CCC(NC(=O)C=CC3CCCC3)C2)=O)CCc2nncn2C1 N1(C(C2(C#N)CCCC2)=O)CCC(C2CCN(C(=O)C(F)(F)c3nccs3)C2)C1 C#CC1CN(C(C2CC3(CCC3)C2)=O)CCN1C(=O)CCc1cnc(C)s1 C1(CNC(CN(C(C2C(CCOC)C2)=O)CC2CC2)=O)CC2CCC1O2 c1(OCC)nc(C(N2CCCC2C(C)NC(=O)C(C)Cc2ccccn2)=O)co1 CN(OCC(F)(F)F)C(=O)CC(=O)N(C)CCc1ccccc1 N1(C(CC(CC)C2CC2)=O)CC2CC1CN2C(C12CCC(C1)OC2C)=O C(=O)(C(F)(F)C(F)(F)F)NC1CC(C)(CNC(CC(CCC)c2ccccc2)=O)C1 C1(C(=O)OCC(C(C)=O)=O)C2CC(C(O)C2O)S1(=O)=O c1(C(N(CCN(C(=O)C(C)C#N)CC)CC)=O)cc(C)cc(C)c1O C1(CCC)CN(C(C2CC(O)CN2C)=O)CCN1C(c1nc(Cl)sc1C)=O c1(NC(NNC(=O)c2ncn(C)c2)=O)ccc(CS(C)=O)cc1F CCCC(CC)CCC(=O)N(C(C)C(=O)Nc1cc(C)cc(C)c1O)CC N1(C(c2c(C)nc(CC)o2)=O)CCCC(NC(=O)Cc2cc(CC)nn2C)C1C c1(OCC(C)C)ncc(C(=O)N(CCN(C(=O)C(C)O)C)C2CC2)cc1Cl Cc1cc(C=CC(N2CC(CNC(c3cn(C)cn3)=O)C(C)C2)=O)on1 C1(NC(C(CC)(C)F)=O)COC2(C1)CN(C(c1cc(C(C)(C)C)n[nH]1)=O)C2 c1(C(N(C)CC2(NC(C3COCCC3(F)F)=O)CC2)=O)ccc2cccnn12 C1(NC(c2snc(O)c2Cl)=O)CC2CCC1N(C(=O)C1=CCCCC1)C2 N1(C(c2ccc(-c3ccncc3)o2)=O)CC(C2CN(C(c3cnc[nH]3)=O)C2)C1 N1(C(CCC(=O)NCC)=O)CC(NC(C2CC2c2cccs2)=O)CC2(CCC2)C1 N(C(=NCCc1sccc1Br)NCC1CC(C)(F)C1)CC(C)(C)C c1(CC(=O)NCC(CNC(c2c(C)nco2)=O)C(F)(F)F)nc2c([nH]1)CCCC2 CC(C)C(C(=O)NCCN(C)C(c1cn(C)nc1C1CCCCC1)=O)NC=O c1(CNC(C2(CCNC(C3(CC#C)CCCO3)=O)CCC2)=O)ccc(Cl)cn1 CCCCC(C(=O)NCC1(C)CCCS1)NC(c1sncc1CC)=O N1(C(CCOCCCOC)=O)CCCC(NC(c2cccnc2C(F)F)=O)C1C C1(C(=O)NC(CNC(c2ccc(C(C)=O)o2)=O)(C)C)Cc2cc(C)c(C)cc2O1 c1(OCC)nc(N2CCC(N(C(=O)CN3CCNC(=O)C3)C)CC2)cc(C)n1 N1(C(C2(CC)CCC2)=O)CC2(C(=O)NC(c3cncnc3)C)CCC1CC2 C(=O)(C1=CCSC(O)C1)NC(C1CCCN1C(c1cnc(O)n1C)=O)C c1(C(=O)NC2CC(NC(c3cnoc3)=O)C2)cc(C2CCCCC2)on1 Cc1nc(=NCC2CC(C)N(C(=O)CSC3CCCCO3)C2)s[nH]1 c1(SC)nc(O)c(C(N2CC(CNC(c3cc(Br)n[nH]3)=O)CC2C)=O)cc1C#N c1(C(=O)NCC2CCN(C(C=C(CC)C)=O)C23CC3)ccc2c(ccn2C)c1 c1(C(CNC(c2c(CC)csc2)=O)NC(c2cnsc2)=O)cccc(C)c1 N1(C(CCC=CCC=C)=O)CC(CCNC(c2cnn[nH]2)=O)C(C)C1 C1(NC(c2nc(CC)sc2)=O)C2CCN(C(=O)CCOC)CC12 C1(C(=O)NCCNC(c2cccc(SCC)c2)=O)CCCCNC1=O N1(C(c2c(C)noc2C(F)(F)F)=O)CC2CCC1CN2c1nc(Cl)ncc1Br C1(NC(Cc2cnc(C)o2)=O)CN(C(=O)CNc2ccccc2)CC1C CN1CCN(C(=O)CCc2ccc(Cl)c(F)c2)CC1CNC(=O)Cn1ncnn1 C1(C(=O)NC2CCN(C(N)=O)C2)CCCCN1C(=O)C=CC1CCOCC1 N1(C(Cc2c(C)nn(CC(C)C)c2C)=O)CC(NC(=O)CC(C)O)C2(CCC2)C1 CC1CC(NC(=O)Cc2cc(C3CC3)nn2C)CN(C(=O)Cc2cnn(C)c2)C1 C(=O)(C(F)CC(C)(C)NC(C1CC2(CC(=O)C2)C1)=O)NCCCC1CC(C)C1 N1(C(CCSCCCC)=O)CCN(C(C(=O)NCCCC2CC2)C2CCOC2)CC1 c1(CNC(=O)NC(C#CC#C)(C)C)cccc2c1CCC2 C(CNC(c1cc(C(N)=O)co1)=O)(C(=O)NOCCC(F)F)OC C1(C)(C(=O)NC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CCNC(=O)C1 C1(C(=O)NCCC2CC(NC(c3c(CC)[nH]nc3Cl)=O)C2)CC1C1CCCC1 C12(C(=O)NC34CC(C3)N(C(=O)CSCC3CCCCO3)C4)CCC(CC1)C2 c1(NC(C2C3CN(Cc4ccnc(OC)n4)CC32)=O)cc2ccccc2nc1Cl C1(CNC(c2c(C)snc2)=O)N(C(=O)C=Cc2cncc(O)c2)CCCC1(C)C N1(c2cn(C)nc2)CCC(NC(=O)CN2CC(C3(C(=O)N)CC3)C2)C1=O.C(=O)O N1(CCN(C(=O)CC2CC=CC2)C)CCN(C(C2CSCC(=O)N2)=O)CC1 c1(C(N2C(CNC(=O)CN3CCOCC3)C=CC2)=O)cc2cc(F)c(F)cc2[nH]1 c1(CNC(CN(C2CCSC2)C)=O)cc(C(F)(F)F)ccc1Br c1(C(=O)NCCCC(C)(C)NC(C(CC)=CC)=O)c(O)cc(=O)n2c1CCCC2 O=C1CCc2cc(CNC3CCN(C(C4(c5ccc(F)cc5)CC4)=O)C3)ccc21 c1(C(=O)NC2CCC(N(C(c3cc(CC)no3)=O)C)C2)cnccc1C C1(C(=O)NC(CNC(COC2(C#C)COC2)=O)C2CC2)(CCC)CCNC1=O C1(C(=O)OCC)CCCC(NCCN(CC(=O)NCCCSC)C)C1.C(CO)O C(CCC(C(=O)NCc1cc(OC)ccn1)NC(=O)CN1CC2CC2C1)OC CC(C#N)CS(=O)(=O)N(C(C)(C)C(=O)OC(C)(C)C)C1CC1 C12(NC(CCC=C(C)C)=O)COC(CNC(c3c(C)coc3C)=O)(C1)C2 N1(C(C(=O)NCCS(CC)=O)=O)CCS(=O)C(C)C1 C(=O)(C(C)C(O)CC)N1CCC(CC#C)(C(=O)NCC2CCC2CO)C1 C1(C(N2C3C(CNC(c4c(CC)cccc4)=O)C(C3)C2)=O)Cc2ccccc2N1 CCC(CC)(CC)C(=O)N1CCN(C(c2cn(C)cn2)=O)C(C2CCC2)C1 c1(C(=O)NCC(CNC(Cc2n(C)nnc2)=O)(C)O)ccncc1N C(C(C)(C(C)C)C(C)C)NC(C1OCCC(NC(CCC(=O)NC)=O)C1)=O CC(CCC(C)(C)C)C(=O)N1CC(OCC(=O)OC(C)(C)C)C1 N1(c2nc(C(F)(F)F)cc(C)n2)CCC2(CC1)CC(NC(=O)CC(C)C)CO2 Nc1sc2c(c1C(N1CCOC(CCNC(=O)C(F)=C3CCC3)C1)=O)CCSC2 C1(C(N(C)Cc2cn(CC)nn2)=O)(CNC(C)=O)CC12CCC2.C1(=O)CC1=O C1(C(=O)NC(C=C)(C)C)CN(C(C2CC23CCOCC3)=O)CC1C1CC1 C1(CN(C(C2CCCN2S(C)(=O)=O)=O)CC)CCCN1C(c1cc(C)c[nH]1)=O CCC(C(=O)NCC1(C)CCN(C(=O)C(CC2CCC2)OC)CC1)C(C)(F)F Cc1nc(C)c(C(=O)NCC(C)N(C(=O)CCC23CC(CO2)C3)C)nc1C CN=c1[nH]c(=NCCCSc2cccc(F)c2)[nH]c(=NCCC2CCCC2O)[nH]1 CC1CN(C(C23CCCN2CCC3)=O)CC1(C)C(=O)NC1CCCCC1(C)C c1(N(CCS(=O)(=O)NC)C)nc(N2CCC(C)(F)C2)c2cnn(C)c2n1 C(C(C(=O)NCC(C)Cc1cn[nH]c1)C(C)(C)C)NC(CSCCCC)=O C1(C(=O)NC2CC(C)(OC)C2)CCC2CC1CO2.C(C(F)(F)F)NC(CN(C)C=O)=O C(CN=C(NCCN(C)C)NCC(C)Sc1cn(C)nc1OC)OCC c1(C(N2C3CN(C(Cc4c[nH]c(=N)[nH]4)=O)C(CC3)C2)=O)cc(=O)n2nccc2[nH]1 Cn1[nH]c(=NC(=O)C(O)CCNC(C2CCCN2C)=O)cc1C(N)=O C=CCN(OC)C(C)=CC1CCCN1C(=O)C=Cc1cncn1C C1(NC(C(C2CCCC2)OCC)=O)CCN(C(c2cnc(=N)[nH]c2)=O)CC(O)C1 c1(C(N2CC3C(NC(c4ccoc4C(F)(F)F)=O)C3C2)=O)cc([N+](=O)[O-])n[nH]1 C1(NC(C)=O)CCC(C(=O)NCC(C2CC2)NC(=O)CSC2CCCCO2)CC1 CC(CN=c1[nH]c(NC2CCCc3nn(C)cc32)nc2c1CCCC2)C(F)F C1(C(=O)NC2CC2)C2CC3C(C2=O)C13.C12(C)CCN(C1)C(=O)C1CC1C(=O)NC2C.CF Cc1ncc(C(N2CCC(N(C(=O)Cc3cnccc3Cl)C)C2)=O)n1C N1(C(CCCC)=O)CCC2(CC(C(=O)NCCCc3ncc[nH]3)C2)C1 CC(C)CC(C(=O)NOCC(=O)Nc1ccncc1)C(C)C N1(C(=O)NC(C(CC)CCN)C)CCC2(CCCC(C(=O)OC(C)(C)C)O2)CC1 O=C(C1Cc2ccc(F)cc21)NCC1C=CCN1C(c1cc(C2CC2)no1)=O C1(COC)(NC(=O)NC)COC1.C1(C)CNC(=O)N1.C(C)(C)(C)O N1(C(C(C)CO)=O)CC2CN(C(C3CC3c3ccncc3Cl)=O)CC2C1 Cc1ccc(C2(C(=O)NCC(C)(C)CCNC(C3NC(=O)OC3C)=O)CC2)cc1 C1(C(N(CC(C)(C)NC(C(F)=CCC)=O)C)=O)C2CC3CC(C2)CC1C3 CCCC(C)C(C)NC(=O)COc1ccc(OC)cc1 C(=O)(CCC(C)C)NC(C)Cn1cc(CCC(c2nnc(C)o2)C)nn1 Cc1nc(C)c(CCC(N2CCN(C(C34CC(F)C3C4)=O)C(CO)C2)=O)c(O)n1 C12(C(=O)NC(=O)CCN3CCC3)CCC(NCCC3C=CCC3)(CC1)CC2 CC1(C)CC(C(=O)NCCC2(C(=O)NCCCF)CC2)C1 N1(CC)CCOC(C(=O)N(C)CC2CN(C(=O)C(C)C(C)O)CCO2)C1 CC(=O)CC(C)(C)C(=O)N1CC2CC(C(=O)NCC3CC4CCC3C4)C(C2)C1 C12(C(=O)NCC3N(C(CCCCC)=O)CC4CC43)CCC(OC)(CC1)CC2 C(C(C(=O)NCCn1cc(C)cn1)NC(c1cc(CC)no1)=O)OCC C(=O)(C(=O)C(C)(C)CC)NC(C(N1C(CC#C)CCCC1)=O)C C1(C)(N(C)C)CCN(C(=O)CCC2CCCN(C(c3ccc(F)nc3)=O)C2)C1 c1(CC(N2CCC(C(F)(F)F)(CO)CC2)=O)c(F)cc(F)cc1F CCCCC(CC)C(=O)N1CCCCC(C(N2CC(O)(CC)C2)=O)C1 CC1C(NC(C2(C)CC2(C)C)=O)CC2CCC1N2C(c1c(F)cccc1F)=O C1(C(=O)NC(CCCNC(C(CC)SC)=O)C)CC1C1CCCCC1 N1(C(c2ccccc2-c2cccc(C)c2)COC)CCC2(CC1)CNS(=O)(=O)N2C Cc1cccnc1C(=O)NOC(C)(CO)C(=O)NC1CCCC(C)C1 N1(CC(N2CC(S(=O)(=O)N3CCOCC3)C2)C)CCC2CCCCC12 N1(CC)CCC(CC2CCCN2C(=O)Cn2[nH]cnc2=N)CC1 c1(CN2C(C(=O)Nc3cccc(F)c3O)CSCC2)cc2ccccc2s1 N1(C(C(C)O)=O)CCCCC1C1CCCN(C(=O)CC2(C)CC2(Cl)Cl)C1 C(CC(CO)NC(c1cc(CNC(=O)CCN2CCCCC2)on1)=O)=CC c1(C(N2CC(C)(CCC(=O)N(CC(C)CO)C)C2)=O)ncncc1N c1(C(N2CC3C(C(N4CC5COCC5C4)=O)C3C2)=O)nc2cccc(Cl)c2s1 c1(C(C)NC(C)CNC(c2cc(O)nc(C3CC3)n2)=O)cccc2oc(C)nc12 C1(NC(CC=C(C)C)=O)CN(C(=O)C=C(C)C2CCCCC2)CC1(C)C C1(NC(c2cnc[nH]2)=O)CCC12CCN(C(=O)C=Cc1ccccc1)CC2 C(=O)(CCC(C)(C)C)N1CC(C)C(NC(c2cccc(I)c2)=O)C1 C1(NC(c2cn(CC)nn2)=O)(CO)CCCN(C(=O)CC2COCCO2)C1 c1(NC(C2CC(CNC(C3CC(C(C)(C)O)C3)=O)C2)=O)ccc(CO)cn1 N1(C(C=Cc2c(C)noc2C)=O)CC2CCC(C1)N2C(C12CCC(N(C)C)C1C2)=O Cc1nocc1CC(N1CCCC1CCC(=O)N1CC(c2ncccn2)C1)=O N1(C(C(n2cc(Br)cn2)C)=O)CC2C(C(N3CC(F)C3)=O)C2C1 Cc1n[nH]c(C)c1CCCNC(=O)NCC1CC(NC(=O)OC(C)(C)C)C1 N1(C(c2c(OC)ccs2)=O)CCC2(CC1)CC2NC(c1c(SC)cccc1F)=O C1(C(N2CC(NC(C3(c4ccsc4)CC3)=O)C3(CC3)C2)=O)CCc2nc[nH]c2C1 c1(-c2cn(CC(C)NC(C3CN4CCC3C4)=O)nn2)c(C)nn(C)c1C C1(C(=O)NC(CCCC)CNC(=O)C(CO)SC(C)C)CCS(=O)(=O)CC1 CC1CN(C(c2cc(Cl)cs2)=O)C(C)CN1C(C1CC1C(F)(F)F)=O Cc1ccc2oc(=NCC3CN(C(c4cc(C(C)(C)C)no4)=O)CC3C)[nH]c2c1 c1(CNC(CN(CCC)C)=O)n[nH]c2c1CN(C(c1cc(N)cc(O)n1)=O)CC2 N1(CCNCC2CCC2)CCC2CC(C(=O)NC3CCNC3=O)C2C1 C1(NC(C2(SC)CN(C(c3cc(C)c(C)s3)=O)C2)=O)CCC(F)(F)C1 C(C(CC(=O)N1CC2CC1C2NC(c1nccc2[nH]ccc12)=O)C(F)F)N(C)C N1(CC)CCCN(C(=O)CCn2cc(CCC(C3(O)CCOC3)=O)nn2)CC1 N1(C(=O)NCCCl)CCC2CN(C(c3c(Cl)cc(Cl)cc3Cl)=O)CC2C1 N1(C(C2CN(C(c3c(C)con3)=O)C2)=O)C(C)CCCC1C.C12CSCN1C2=O C1(C(=O)NC(CC=C)(C)C)CC2CC1CN(C(=O)C(C)CSC)C2 CCC(CC)(CC(=O)OC)C(=O)N1CC(NC(c2ccc3c(c2)CCCO3)=O)C1 C(=O)(CS(=O)(=O)CC1CCCO1)OCC1(OC(C)C)CCOCC1 C1(NC(C(C2CCN(C(CC(=O)NCC)=O)CC2)C)=O)CC2COCC(C1)C2 C(=O)(C(F)(F)C(C)O)N(C)CC1CCN(C(C(C)n2cccc2)=O)CC1 N1(C(CCC(CC)NC(c2c(C)cccc2O)=O)=O)CCn2ncc(O)c2C1 c1(OC)ccc2c(c1)C=C(C(=O)N1CCC(O)(CN(C)C(C3CC3C)=O)C1)CO2 c1(-c2cn(CCCN(C)C)nc2)ccnc(C(=O)NCc2cocn2)c1 C1(NC(C(C)(C)OCC)=O)CN(C(C2(Cc3cccs3)CC2)=O)C2(CCCC2)C1 c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(C2CCCC2)OC)CO)c(Cl)c1 C(CC(Cc1ccccc1)N=c1nc(-c2ccccc2)o[nH]1)SCC c1(NC(CC(C)NC(C(COCC)(C)C)=O)C)ncc(C(=O)OC)cc1Cl c1(CC(=O)NC2CCC(NC(C)=O)CC2)ccc(C)cc1Br CC1CN(C(C2(C)C=CCC2)=O)CCC12CCN(C(=O)CC(C)(C)C(F)F)CC2 N1(C(C(CNC(c2c(N)nccn2)=O)CC2CC2)=O)CC2C=CC1CC2 C(CCCCNC(=O)C(=O)NC1CC1)N(CC(C)N(C)C)C Cc1ccccc1C1CC(OC(F)F)C1.C(=O)(C(C)(C)CO)N1CCC1 c1(OCC(=O)NCC2(CCNC(C(C)(C)C3CCC3)=O)CC2)ccc(Cl)nc1.COC c1(C(N2CC3C(C(=O)NCc4cn(CC)nc4)(C3)C2)=O)ccc2c(c1)NCCO2 c1(CN=[N+]=[N-])ccccc1NC(C1CC(F)CN1C(c1cccs1)=O)=O c1(C(=O)NC(CNC(C2N(C(=O)OCC)CSC2)=O)C)cc(Cl)c(Cl)cc1C C1(C(=O)NC2CC(C)C2)CN(C(c2ccnc(SC(C)(C)C)c2)=O)CCC1C C1(NC(COCC)=O)COC2(CCCN(C(=O)C(=O)NOC)C2)C1 C1(C(N2CCN(C)CC2CNC(=O)CSCC(N)=O)=O)CCCC12CCOCC2 Cc1cc(F)ccc1C(N1CC(O)CCC1C(=O)NC(C)(C)CCF)=O Cc1ccc2cc(C(=O)NC3CCC(NC(c4[nH]nnc4C)=O)C3)ccc2c1 c1(C2(C(=O)NCC3CCN(C(C(C4CCOCC4)=O)=O)C3)CC2)ccc(O)cc1 C1(CC)CN(C(=O)CCCOC)CCC1NC(c1cc(C(N)=O)[nH]n1)=O c1(C(=O)NC2CCC(CNC(=O)CCc3ncc[nH]3)C2)c[nH]c2cc(O)ccc12 CC1COCC(C(=O)NCC2CCN(C(=O)Cc3cnn(C(F)F)c3)CC2)O1 O1N(C)C(=O)C2(CC2)C(C)NC(=O)C1.C1(CC)CCC(=O)C1 C1(NC(Cc2c(C)non2)=O)CC2CC(C1)N(c1nc3ccccc3o1)C2 Cc1cc(C(=O)NC2C3CCN(C(=O)Cc4cccs4)C23)cnc1C(F)F C(CC(C(=O)NC1CCCC1)NC(c1ccnnc1C)=O)OC c1(CN(CF)CCl)cc2c(nc1Cl)CCS(=O)(=O)C2 N1(C(c2nc(C)oc2)=O)CC(NC(C23CSCC2C3)=O)CC12CCC2 N1(Cc2cnn(C)n2)CC(NC(c2ccc(F)c(C(F)(F)F)c2)=O)C(C)(C)C1 N1(C(C2C(C)C2(F)F)=O)CCC(C)(CNC(c2cc(C(N)=O)cn2C)=O)CC1 C1(CNC(c2c(CC)c[nH]c2)=O)CC(F)(F)CN1C(c1ccc(C)c(Cl)c1)=O c1(C(=O)NC2C=CC(CNC(C(C(C)(C)C)O)=O)C2)ccc2cccnc2n1 N1(C(C(CO)N(C)C)=O)CCC(C2CN(C(=O)COc3cccc(F)c3)C2)CC1 C1(C(N(CC(C)NC(c2cc(C(F)(F)F)c[nH]2)=O)C)=O)CCC(C(=O)OC)C1 N1(Cc2cc(C#N)on2)CCc2n[nH]cc2C1.N12CCCC1C=CC2=O c1(C(=O)NCCCN(C(C(CC)N(C)C)=O)CC)cc(Br)n2c1CCC2 C1(NC(c2ccc(CCC)cc2)=O)CC2(CCC1NC(=O)CC1CC1CC)CC2 c1(C(N(C(=O)CCNC(C2CCC2CC2CC2)=O)CC)=O)cn(CCN)cn1 C1(NC(c2cccc(N(C)C)c2)=O)CC1C1CCCN(C(=O)Cn2cncn2)C1 C1(CC(=O)N(CCN(C(=O)CCc2ncco2)C)C)CCC(C(F)(F)F)O1 c1(C(=O)NCCCn2cc(-c3cnn(C4CC4)c3)nn2)cc2cc(F)ccc2s1 N1(C(c2c(C(N)=O)cccc2)=O)CCN(C(=O)Cn2cnnc2O)CC1CO c1(C(=O)NC2CCC(F)(CNC(C(C)SC)=O)C2)ccc2c(n1)CCOC2 N1(C(CCC(C)OC)=O)CCN(C(c2ncn(C)n2)=O)C(c2cn[nH]c2)C1 C(c1cc[nH]n1)=CC(N1C(CNC(C2CC(C)C2)=O)CC1)=O C1(OC)(CNC(c2nc(Cl)cs2)=O)CCN(C(C2CC3CCC2O3)=O)C1 c1(C(N2CC(N(C)C(C3C4CCCC34)=O)C(C)(C)C2)=O)[nH]cc2c1CCCC2 Cn1ncc2c(N3CCN4CCCC4C3)nc(=NC3CCCCCCC3F)[nH]c12 CC(C)C(F)C(=O)NC1CCC(CCNC(c2ccc(O)cn2)=O)C1 c1(C(N2CC=CC(NC(C(c3ccccc3)OC)=O)C2)=O)cc(F)ccc1C C(CC(CC)C(=O)N1CCC(N(C(=O)Cc2c(C)cccc2F)C)CC1)=CC C1(CC)C(C(N2CC(CSC)C2)=O)CCN1C(=O)Cn1nc(C)nc1C c1(C(=O)NCC2CC(C)N(C(=O)Cn3nnc(=N)[nH]3)C2)ccc2c(c1)C(=O)NC2 C1(C(=O)NCC(=O)OCC)CCN(C(=O)C(=O)CC(C)C)C12CCC2 c1(-n2c(C(=O)OCc3cccc(N)c3)ccn2)c(F)cc(F)cc1F C(CCC(=O)NCc1nocc1C(=O)NCC1(N(C)C)CCCC1)C1C(C)C1 N1(C(C2(C)CC3CCC2C3)=O)C2CCC1CN(C(c1cnc[nH]1)=O)C2 CC1=NOC2(C1)CC(C(=O)NC1CC1NC(c1nc[nH]c1C(C)(C)C)=O)C2 c1(OC)ccc(C(=O)N(CC(C)NC(=O)C(C2CCOCC2)F)C)c(OC)n1 C1(CC(=O)NCCCC2C(=O)NC(=O)N2)C2CCC(C2)N1C(=O)C=CC1CC1 C1(CCOC)(NC(=O)C(C)Nc2cnn(C3CC3(F)F)c2)CCOC1 C1(NC(=O)CC2COC3CC2C3)(CNC(c2cc[nH]n2)=O)CC2CCC1CC2 N1(C(c2n(C)nc(O)c2)=O)CC2CCC(CNC(c3cc(F)n(C)n3)=O)C2C1 C12(C(N3C(C(=O)NCCCC(C)(C)OC)CSCC3)=O)CCC(C1)OC2C c1(C(N2C(C)CCC(NC(COCCC)=O)C2)=O)cc2cc(Cl)cnc2[nH]1 c1(C(=O)NC(CN(C(=O)C(c2cn(C)nc2C)C)CC)C)cn(C)c(=O)c(C)n1 c1(CC)c[nH]nc1C(=O)NCC(C)C(=O)NCc1cc(O)ns1 CC1(C)C(NC(C2CC(O)C2)=O)CCN1C(=O)CCc1ccc(F)cc1F c1(CC)ccncc1NC(=O)C(CCNC(=O)CCOCCOC)OC c1(OCC(=O)NC2C=CCN(C(C(CCOC)C)=O)C2)c(Cl)cccc1[N+](=O)[O-] c1(CO)ccccc1C(c1nnnn1C)NCC1(c2ccccc2)CC(O)C1 C1(N=[N+]=[N-])(C(=O)Nc2c(OC)cccc2)CCN(C(c2ccc(O)cc2F)=O)C1 C(=O)(C#CC(C)C)N1CC(CC(CNC(Cc2snc(C)n2)=O)(C)C)C1 c1(C(N2CCC(CO)C(F)C2)=O)ccc(-c2ccccc2C2CC2)c(Cl)c1 N1(C(C2C(CC)N(C)CC2)=O)CCN(C(c2cccc(C3CC3)n2)=O)CCC1C c1(C(=O)NCC2N(C(c3n(C(C)C)ncc3Cl)=O)CCC2)ccc(Cl)nc1O N1(C(C2OCCN(C)C2)=O)CCC(C)(C)C1C(=O)Nc1ccc(CN(C)C)cc1 N1(CC(C)C)CCC(O)C(C(=O)NCC2(C)CC(CO)C2)C1 C1(C(=O)NC2C(CNC(CCn3ncc(C)c3)=O)CCC2)(CCF)CCOCC1 Cc1ccc(F)c(CC(N2CCC(CO)(NC(=O)C3=CC(C)(C)C3)C2)=O)c1 C1(CCNC(c2c(C)scc2)=O)CC(F)(F)CN1C(=O)C=Cc1cncc(O)c1 CN1C(=O)CC(NC(C2CC(O)CN2C(=O)CCc2nncn2C)=O)C1=O c1(C(C)NC(=O)NCC2CCCC2C)ccnc(N(C)C)c1 c1(C(=O)NC2CCCN(C(c3cc(C)c(F)cc3)=O)CC2)ccn2nccc2n1 S(=O)(=O)(c1c[nH]c2cccc(Br)c12)NC(C(=O)OC)CSC N1(C(Cc2nc(C)oc2)=O)CCCC2C1CCCN2C(C1CC(=C2CC2)C1)=O Cc1cc(N2CC3(C2)SCCC3NC(C2CC(C)OC2C)=O)nc(S(C)(=O)=O)n1 N1(C(C(=O)OCC)=O)CCC(NC(=O)C=C(C)c2ccc(OC)cc2)C(C)(C)C1 c1(CC(C)N(C(c2ccccc2N)=O)CCl)ccc(Br)cc1F.CCON CC(C)C(C)CC(=O)N1CCC(O)(Cn2cc(CCC3CCCO3)nn2)C1 S(=O)(=O)(CCCN=c1[nH]c(=NCC(c2ccco2)OC)c2sccc2[nH]1)NC N1(C(C(=O)c2ccco2)=O)CC(N=c2ccnc(Cl)[nH]2)C2(CCC2)C1 CCC(F)(F)CC(=O)N1CCC2(NC(=O)CCSc3ccc(C)cc3C)CC2C1 C1(C(C)NC(C2(C)CC(=C)C2)=O)CN(C(=O)C2=CCCO2)CCO1 C1(NC(c2cccc(CC=C)c2)=O)CCC(C)N(C(=O)CSCCOC)C1 N1(c2cccc(N)n2)CCCC(NC(=O)N(N2CCCC2)Cc2ccc(Br)s2)CC1 c12cccc(c1)C(COC)NC(=O)C(=O)N2.C(=O)(CC(C)C)OC c1(C(=O)NC(C(C)(C)C)CNC(=O)CC2CCCCO2)csc2ccncc12 N1(C(c2ccc(C)cc2N)=O)CCCN(C(C2CCCCO2)=O)C(CO)C1 c1(C(N(CC2N(C(c3c(CC)nn[nH]3)=O)CCC2)CC)=O)c(C(C)C)cnn1C c1(OCC(=O)OCC(=C)OCOC)cc(C)c(F)cc1Br C1(NC(=O)CC2CC3CC3C2)(CO)CCN(C(c2ccc(O)c(Cl)n2)=O)CC1 c1(C(=O)NCC(C2CC2)NC(CSCCOC)=O)c(C(C)C)cccc1F c1(CC)noc(C(=O)NC2CN(C(=O)Cc3ccc(COC)cc3)C2)c1C [N-]=[N+]=Nc1ccccc1C(=O)NCC1(NC(=O)C(F)=CC2CC2)CCCCCC1 Fc1ccccc1Cc1nc(-c2cc[nH]n2)nn1CC1CCC1 N1(C(c2nn(C(C)C)cc2Br)C(=O)NCCSC)Cc2ccc([N+](=O)[O-])cc2C1 C#Cc1cccc(CNC(C2CC(NC(=O)C(C)OCCN(C)C)C2)=O)c1 c1(CNC(c2c(OC)ncnc2OC)=O)c[nH]c2cccnc12 CC(C)C(O)C(C)(C)CNC(=O)CONC(C1CC2CCC2C1)=O CC1(NC(c2csc(Cl)n2)=O)CCN(C(c2ccc(C3CC3)nc2)=O)C1 N1(C(C=C)=O)CCN(CC2CCN(C(c3cnc(C(C)O)s3)=O)CC2)CC1 C1(CC(=O)NC2C(C=C)CN(C(C3CCCCC3)=O)C2)CC2(CCCC2)CO1 CS(=O)(=O)CCCCCNC(=O)C(=O)NC(c1ccc(F)cc1F)C1CC1 Cc1cccc(CC(N2CCCCC(NC(c3ccnnc3O)=O)C2)=O)c1F n1(C2CN(C(C=C(C)Cl)=O)C2)cc(CNC(=O)CC(=O)NC2CC2)nn1 C1(CC(=O)NC2CC(N(C(=O)CSC3CCCC3)C)C2)CCCCC12CC2 N1(C(C(c2cccnc2)NC(c2n(C(C)C)ncc2)=O)=O)CC2(CC2)CC1C N1(c2snc(SC)n2)CCCC(C)(C(=O)NCC2COCC2N(C)C)C1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(N(C(=O)Cc2c(F)cccc2F)C)C(C)C1 C(=O)(CCN=C(NCc1ccc(C(C)C)c(C)n1)NCc1ccc(C#N)s1)NC c1(CNC(C2(COC)CC2)=O)ccc2c(C)c[nH]c2c1.c12noc(C)c1NC2=O Cc1ccc(C(N2CCCC2C(C)NC(C2CCCCCC2)=O)=O)nn1 Cc1c[nH]c(C(N2CCC(CCCNC(C3CC3Cl)=O)CC2)=O)cc1=O C12(NC(C(n3ncc(C)c3)C)=O)CCCC1N(C(c1ccccn1)=O)CCC2 c1(C(=O)NC2(CC)CCCN(C(=O)C=C(C)Cl)C2)cnn2cccc(C)c12 N1(C(c2cccc(SCC#C)c2)=O)CC2CC(NC(C3CCCSS3)=O)CC1C2 C#Cc1ccc(C(=O)NC(CC#CC)C(N2CCCC3(CC2)CC3)=O)c(C)c1 C(C(C)(C)C(=O)NC1CC(C)(CNC(C2(C)CCCC2)=O)C1)NC(C)=O c1(C(N(C)CC2N(C(C3C(OC)CC3)=O)CCC2)=O)cc(C)n(C2CC2)n1 N1(C(C(CC#C)(C)C)=O)CC2CCCC(CNC(=O)C(CC)SC)C2C1 c1(C(=O)NC2CC(NC(c3ccc(C)c(C)c3)=O)C2)cc2c(cc1O)CCC2 C1(NC(C(C)NC(=O)NC)=O)CCN(C(=O)C(c2ccc(F)cc2C)O)CC1C c1(-c2nc(CC(C)(C)C)nn2Cc2ccsc2)ccnc2[nH]cnc12 CC1=CC(C)=NS(=O)(=O)N1CC(N1CCCC1C1CCCOCC1)=O c1(CC(=O)NC2CCN(C(c3ccc(N)cn3)=O)C2)cc(O)cc(Br)c1 c1(C(N2CC3CC2CN3C(C2C(C=C(C)C)C2(C)C)=O)=O)cc2cccnc2nc1O C1(NC(CC)=O)CCN(C(=O)OC(C)(C)C)C1.C12CCC(C1)C(=O)N2 CCC(C)CCC(=O)N1CC2(CC2)CC1CNC(=O)CCc1cccc(F)c1 N1(C(CCCOCCC)=O)CC(NC(=O)C(C)(C)CNC(C)=O)C(C(F)F)C1 CC(C)(CNC(=O)C(c1ccoc1)NC(c1ccns1)=O)CCCO N1(C(c2c(C)ncn2O)=O)CCCC(C2(NC(=O)CO)CC2)C1 C1(C(N2C(C)(C(=O)NCCC(C)N(CCC)C)CCC2)=O)CCC=CCCC1 C12(C(=O)NC3CC(NC(C4CC5C=CC4O5)=O)C3)CCCN1CCC2 C12(CNC(c3c(C)ccnn3)=O)CCCCC1N(C(c1cncnc1C)=O)CC2 c1(C(=O)NC2CC(CNC(C(c3ccnn3C)C)=O)C2)ccnc(C(C)(F)F)c1 c1(NC(c2cc(Br)ccc2C)C(=O)OC)ccc(S(=O)(=O)N(C)C)cc1 c1(CCC)cc(C(=O)NCC2(CNC(c3cc[nH]n3)=O)CC2)nn1C CC1(CC(N2CCC(NC(C3CC3C#N)=O)C2)=O)OCCO1 c1(C(=O)NC(CC(C)NC(c2c(CC)n[nH]c2)=O)C)c[nH]c2ccc(Cl)cc12 C#Cc1cn(C)nc1C(=O)N(C1CCCC1)CCNC(C1(C)CC2C=CC1C2)=O c1(N(C(N(CC)Cc2[nH]ccc2C)=O)CCN2CCOCC2)cccc(CO)n1 Cc1cc(C(=O)NCC=CCC(=O)N(C)C(C)C2CC2)c(C)o1 c1(C(N2CCC3(CN(C(CC(CC)C)=O)C3)C2)=O)ccc([N+](=O)[O-])c(N)n1 O=C(CS(=O)(=O)C1CCCC1)NC1C2CC(O)C1N(C(C1(CO)CCCO1)=O)C2 Cc1cccc(CC(C)(O)C(C)NC(=O)N(C)CCc2ncon2)c1 N1(C(c2c(C)cc(C)s2)=O)CCCN(CCC(=O)NC(=O)CC2CCCC2)CC1 c1(CN2C(C(=O)Nc3c(C(=O)OCC)cc(C)s3)CCC2)cccc2ncoc12 c1(-c2n(CC3C(C)C3)nc(CC3CCCC3)n2)ccc2ccccc2n1 C1(C(N2CCC(C(=O)N3CCCc4nccn43)CC2)=O)C2Cc3cc(F)ccc3C12 N1(C(C2(COCC)CC2)=O)CCCC(F)(CN(C(=O)Cc2cn(C)nc2C)CC)C1 c1(C(=O)NNC(c2cc(C3(C(F)(F)F)CC3)nc(Cl)c2)=O)ccccc1[N+](=O)[O-] c1(N(C2CC(C)OC2)C(c2cnncc2O)=O)cc2nncn2cn1 CC1(C)CC2(CC2C(=O)NC2CCCCC2CNC(=O)Cn2cnccc2=O)C1 N1(C(c2c(CC)nn[nH]2)=O)CCC(O)(CCNC(c2ccc(C3CC3)nc2)=O)C1 C1(C(=O)NCCCN(C)C(c2cncc(O)c2)=O)CCc2nccn2CC1 C(=O)(C(CN=[N+]=[N-])NC(c1cc(CO)on1)=O)NCC(=C)CC C(=O)(C(O)C(C)(C)C)N(C(C)CN(C)C(c1cccc(-n2ccnc2)c1)=O)C C(=O)(CCCCOC)OC.C1(C)C(=O)N1CCCc1nccs1 Cc1ccccc1-c1cccc(C(=O)NCC2C3CN(C(=O)CC(C)O)CC23)c1 C1(NC(c2c(C(C)C)cccc2)=O)CC2CN(C(=O)C(C)C3=CCCC3)CC2C1 N1(C(CC(CC)C2CCC2)=O)CCC2CN(C(C3(CSC)CC3)=O)CCC12 N1(C(C2ON=C(C)C2)=O)CCN(C(=O)CC(C)(C)c2ccc(F)cc2)C2CCC12 C1(C(N2CCN(CC(C)NC(=O)C=CC3CC3)CC2)=O)CCC2(CCOCC2)C1 c1(Nc2cc(NC(CC)C)ncn2)cccc2nc(O)n(C)c12 C=CCC(C)(C)C(=O)NCCC1CCCN(C(c2cc(CCC)oc2C)=O)C1 N1(C(C2C3CCCC23)=O)CCCC2(C1)CN(C(C1CC13CC(O)C3)=O)CCO2 c1(-c2c(COC)cc(F)cc2)ccc2ncc(C3=C(C)CCCC3)n2c1 C(=O)(C(O)CC(C)(C)C)NC(CC)CCC(=O)N1CCC1(CO)CO O=S(=O)(c1ccccc1Cl)NC1CCC2(C1)CN(Cc1cnc(Br)o1)C2 CCCCC(C)C(=O)N(CCCNC(c1[nH]c(C)c(C(N)=O)c1CC)=O)CCO c1(-c2c(C)noc2)cnc(N2CCOCC2)nc1NC(=O)NCc1cc(Br)cs1 c1(C(N2C(CN(C(C(CC)O)=O)C)CCC2)=O)ccn2ccnc2c1 N1(C(C(CC)N(C)C)=O)CCC(C)(C)C(C(=O)NC(c2ccccn2)CO)C1 c1(C(=O)NCC(CNC(=O)CCc2cnc[nH]2)OC)sc(C)nc1CC(C)C C(=O)(CC1=CCN(C(=O)C(C)(C)C(F)(F)F)CC1)NC(CCSCC)C c1(C(=O)Nc2ccnc(-n3cc(C4CC=CCC4)nn3)c2)cnc2ncccn12 c1(OC)cc(N)c(C(N2CC3(C2)CN(C(=O)C(C)CC(C)C)C3)=O)cc1Br C1(F)(C(N2CCC(C(C)(C)O)C2)=O)CCN(C(C2(Cl)CC2(F)F)=O)C1 C1(NC(COCc2ncc(C)o2)=O)CCC2CC1CN2C(c1cncc(N)c1)=O c1(C(N(CCC(C)NC(=O)CC2CCC(=O)O2)C)=O)ccc2ccoc2c1 C1(CNC(C(C)SC)=O)CC2COCC2N1C(c1cc(=N)[nH]n1C)=O c1(N2CC(C)S(=O)(=O)C(C)C2)c([N+](=O)[O-])cnc2ccsc12 CC1=CCCN(N2CC(Cn3ccnc3)C2)C1 c1(C(N2CCCC(NC(c3c(C)occ3)=O)C2)=O)ncc(P(C)(C)=O)cn1 C(=O)(C(F)(F)CC1CCCO1)NCCOC1CCN(C(CC(=O)N(C)C)=O)C1 CC(CCC(=O)NC1CC1)Oc1ccc(CC(N2CN(C(=O)N(C)C)C2)=O)cc1 N1(C(CN(CCC)C)=O)CC2(C)CN(C(c3ccnc(Cl)c3Cl)=O)CC2(C)C1 c1(OC)ccc(F)cc1N1C(=O)NC(CC(C)(F)F)C1=O c1(C(=O)NC2CCN(C(CC(CC)C)=O)C2C(C)(C)C)cccc(C)c1C CC(C)(C(=O)NCC1(O)CCCC1)C1=CCN(C(=O)CCCCCF)C1 Cc1nc(C(=O)N(C)C(c2cn(CCCCF)nn2)C)c(C)s1 N1(c2cc3nnc(C)n3cn2)CCCC12CCN(C(=O)OC(C)(C)C)CC2 C1(C(=O)NCc2ccc(CC)s2)CCC2CCC1N2C(C1CC(C)(C)CO1)=O CC(C(=O)NCC1(C)CCN(C(c2cnoc2C2CCC2)=O)C1)C(F)(F)C(F)F c1(OC)cnc(Cl)cc1C(=O)NC1CCN(C(c2[nH]c(C)nc2C)=O)C1C(C)C c1(C(N(C2CCN(C(C3CC4CC3C4)=O)C2)CC)=O)csc2c1CCCC2 C(=O)(C(CCC1OCCO1)N1CCSCC1CO)NC(c1ccccc1)CC N1(C(c2ccc(Cl)cc2)=O)CC2CC(C1)N(C(=O)C1=CC(O)CCC1)C2 N1(C(c2c(Cl)nsc2Cl)=O)CCCCC1CNC(C1CC(O)(C(F)(F)F)C1)=O N1(C(C(CCC=C)NC(C2CCCCN2C)=O)=O)CC2(C)CCC2(C)C1 N1(C(c2c(C)nn(C)c2)=O)CCN(C(C2CCOC2C)=O)C(CC(F)F)C1 C1(CNC(Cn2cc(CC)nn2)=O)CCC2(CN(C(=O)Cc3ccon3)C2)O1 CCCC(C(C)(C)C)NC(C1CC(=O)CN1C(=O)COCc1nc[nH]n1)=O N1(C(C2CN(C(C)=O)C2)=O)CCCN(C(=O)CC2(C(F)(F)F)SCCS2)CC1 c1(C(=O)NCC2N(C(C3C(C(C)O)C3)=O)CCCC2)cc(N)c(O)c(F)c1 c1(C(=O)NCC(CC)NC(c2cn(CC)cn2)=O)c[nH]cc(Cl)c1=O c1(SC)ncc(C(=O)NC2CCC(NC(=O)C(C)Cn3ccnc3)CC2)c(O)n1 c1(C(=O)NC2C=CCN(C(=O)COC3CC3)C2)cc(Cl)nn1-c1ncccc1Cl C1(C(N(C(C)CNC(=O)COCCOC)CC)=O)CCCOC1C CC1(C2CCCN(C(c3csc(C#N)c3)C(=O)NC3CCC3)C2)CC1 c1(NC(=O)Nc2nc(C)n(C)c2C#N)ccc([N+](=O)[O-])c(Br)c1 CC#CCC1C(=O)N1.C1(C(=O)N(C(C)COCC)C)C2C3CCC(C3)C12 C#CCC(C(=O)NCc1ncccc1COC)NC(=O)Cn1c(O)nnc1O c1(CONC(c2cc(CNC(CCN(CCC)C)=O)sc2)=O)ccc(O)cc1 CCC(CC)(CO)C(=O)NCC(=O)NC12CC(NC(C3CCCC4(CC4)C3)=O)(C1)C2 CCC(O)C(F)(F)C(=O)NC(CCCNC(=O)CCCC(C)(C)C)C(C)C CC1=C(C(=O)NCC2(NC(=O)CN(C)C(N)=O)CCCCCC2)CCO1 c1(C(CC)NC(CN(CC(C)C)C(C)=O)=O)ccc(-c2ccncc2)o1 c1(NC(CSCCNC(C2(C)C(CC)CCC2)=O)=O)cc(C)nnc1O C1(Cc2ccc(-c3nc(C)on3)cc2)CCCC1C1CC1.C12CCCC1NC2=O N1(CC2OCC(C(C(=O)OC)(C)O)C2)CCC(c2ccccc2)CC1C C(=O)(C1=CCCCCC1)NCCC1CC(NC(C2(C)CCC(=O)N2)=O)C1 C1(C(N2CCC(C)C2CNC(=O)CC2(O)COC(C)(C)C2)=O)CC12CCCCC2 N1(C(C2CC(CC)C2)=O)CCCCC1CN(C(=O)C(C1CCOCC1)C)C CCCCC(C)C(=O)NC1CC2(C1)CC(NC(=O)CC1CC3(CC3)CO1)C2 c1(C(=O)OCCNC(C(=O)N(CC(=C)C)C)=O)cccc(CC)c1 N1(C(C(CC)NC(C)=O)=O)CCOC(CNC(c2cnoc2CCC(C)C)=O)C1 C(=O)(C1CCCc2cccnc21)NC(CCOC)CNC(c1cc(C#N)no1)=O Cc1ccc(-c2ccc(F)cc2Cl)cc1S(N)(=O)=O c1(C(=O)NCC(CO)NC(c2cn(CC)nc2)=O)c(C)noc1N CCCCC(CCC)NCc1ccc(C)cn1.C12CCN(C1)CC2=O C=C1CC(C(=O)N(CC(=O)NCC)C)(CNC(=O)Cc2nc(C)cs2)C1 c1(OCC)ccccc1N1CCN(C(C(=O)NC2CCCC2)c2cn[nH]c2)CC1 CC(C)CC(C(=O)C(=O)C(C)C1CC1)NC(N1CCC(NC(N)=O)CC1)=O C(N=c1nc(N2CCC3(CC2)CC3(F)F)c2c([nH]1)COC2)c1c(Cl)cccc1 C1(CNC(c2ccc(OCC)cc2)=O)CC2CCC(C1)N2C(c1cnnn1C)=O CC(CNC(=O)C(C)CCN(C)C)CC(=O)N1OC2CC1C(O)C2O c1(C(C2CCN2)N(C(C(=O)NC)=O)C)ccc(C)c2ccccc12 CCC(C)(C)C(O)C(=O)NC1(CF)CCN(C(=O)Cc2ccc(C(=O)OC)cc2)C1 c1(C(c2ccn(C)n2)NC(=O)C(c2nncn2C)NC)ccccc1O n1(CNC(C)Cc2ccoc2)c(-c2cnccn2)csc1=Nc1ccc(Cl)cc1 C1(C(N2CCC(CCOC)(NC(=O)C3=C(C)OCC3)C2)=O)CCCC12OCCO2 C1(CCC(=O)NCCN(C(=O)C(=O)Nc2ccccc2)C2CC2)NC(=O)NC1=O c1(C2N(C(C(n3ccc(C4CC4)n3)C)=O)CCSC2)cc(F)cc(Br)c1 N1(C(C(C(C)C)O)=O)CCC12CCN(C(=O)CN1CCCC1)CC2 c1(-c2ccnc(N(C(CN3CCCOC(C)C3)=O)C)n2)csc2cccc(F)c12.C1(C)CC1 CC(C)C(O)C(C)C(=O)NC1(C)CN(C(c2ccnc(C(F)(F)F)c2N)=O)C1 CN1CC(C(=O)NCC2(C)CCCN2C(=O)Cc2c[nH]ccc2=O)NC1=O N#Cc1cnc(NCCC2CCN(C(=O)OC(C)(C)C)CC2(F)F)c(F)c1 C(C)(C(=O)NC(C(=O)N(C1CC=CC1)C)C1(O)CCC1)OCC#C c1(C(N2C(C(N)=O)CC2)=O)coc(CNC(=O)CCC2CCCCO2)c1 c1(C(=O)NCCCSCC2CCOCC2)cnc(CCCO)o1 c1(C(C(=O)NC2(CF)CCN(C(c3cccs3)=O)C2)O)ccc(F)c(Br)c1 c1(OC)cc(C)cc(C(N2CCC(NC(=O)CN(C)S(N)(=O)=O)C(C)C2)=O)c1C c1(CC=C)cccc(C(=O)NCCC2CC(OC)CN2C(=O)CCCCOC)c1 c1(NC(C(=O)N(CCC=C)Cc2cccc(Cl)c2)=O)nc(C)n2c1CCCC2 C(C1CCCn2cc(C)nc21)NC(c1cccc(C2CC2)c1)c1n(CC)nnn1 c1(OCC#C)ncccc1C(=O)NCC(C)NC(c1cccc(CS(C)=O)c1)=O C1(C(=O)NCC2(C)CCCN2C(=O)CC2CCCC2)COC2COCC12 C1(NC(c2ccn(CCOC)n2)=O)CCC(NC(=O)CC2CCCC(=O)N2)CC1 C12C(C1(C)C)CNC(=O)c1cc(no1)C(=O)N2.c1(COC(C)(C)C)ccccc1 CCCC(C)CC(=O)NCC1CCC(NC(=O)C=CCN2CCOCC2)C1 Cc1cc(C(=O)NC2CCC(CC(=O)N(C3CCSCC3)C)CC2)cc(C)c1 N1(C(c2ccc(C)o2)=O)CCC2OCCN(C(C3CCCC3O)=O)C2C1 c1(NCc2cncc(C)n2)ccccc1C(N)C(C)C Cc1sc(-c2ccco2)nc1C(=O)NC1CCC1CNC(C1CC=CC1)=O N1(C(c2cc(OC)n[nH]2)=O)CCCC(O)(CN(C(=O)Cc2cc[nH]n2)C)C1 C1(N(C(c2conc2CC)C(=O)NCCOC)C)CCN(C)C1=O c1(C(N(CCNC(c2cc(OC)c(Cl)s2)=O)C2CC2)=O)cccc(C2CC2)c1Cl Cn1nc(C(=O)NC23CC(CNC(=O)C=CCO)(C2)C3)cc1-c1ccc(F)cc1 CCC(C)(COC)C(=O)NCCCOCCN(C)C(c1ncc[nH]c1=O)=O c1(OCCOC2CCN(C(c3cnc(=N)[nH]c3)=O)C2)cc(NC(COC)=O)ccn1 C(=O)(N=c1cc[nH]c(C)c1Cl)NCCS(CC)=O O=C1CCC(CCC(=O)NCC2(O)CCN(C(=O)CC3COCCO3)CC2)=NN1 C1(NC(C2(C)CCN(C(C(C(C)C)NC(C)=O)=O)C2)=O)CCNC(=O)CC1 c1(C(=O)NC(C)C(=O)NCC2CCSC2)ccc(=N)[nH]n1 c12cc(on1)CCNC2.N1(C(=O)NCC)CC(NC(=O)OC(C)(C)C)C1 C1(C(N2CC(N(C)CC3CC3)C2)=O)CCN(C(C2CC(=O)N2)=O)C12CCC2 N1(C(C(C=C)(C)CCOC)=O)CCCC(C2CC2NC(=O)CC(=O)N(C)C)C1 CC(C)(C)CC(=O)NCCC1CCCN1C(c1ccc(C(N)=O)s1)=O c12ncc(cc1Cl)C(=O)NCC1CCCC1NC(=O)CCN2.Cn1nnc(=N)[nH]1 c1(N2CCC(COC)(NC(=O)CCC3CCC(C)O3)CC2)ncccc1[N+](=O)[O-] c1(C(=O)NC(CCOC)CNC(c2ccc(C)s2)=O)c(SC)cccc1F N1(C(C=Cc2cc(C)no2)=O)C(C)CN(C(c2nn(C)nc2C)=O)CC1C O=S(=O)(c1cncs1)NCc1ccc2c(c1)CC2 N1(C(C(F)=CCC)=O)CC2CCC(C(=O)NC(C3(O)CCCCC3)C)(C2)C1 Cc1nc(NC(C2CCCN(C(=O)CC(C)(C)O)C2)=O)c(F)c(Cl)n1 C(=O)(C#CC(C)(C)CNC(=O)C(C)C(F)F)NC(CCOC)(C)C N1(C(C(C)Cc2ccco2)=O)CC2CC(O)C1C2NC(c1ccc(N)cn1)=O c1(CC)ccc(C(=O)N(C)CC2CN(C(C3CNC(=O)C3)=O)CCO2)cn1 CC1C(C)N(C(C2CC(=C3CCC3)C2)=O)CCN1C(c1coc(CC2CC2)n1)=O N1(C(C(C(C)C)NC(C)=O)=O)CCC2CN(C(c3cc(Cl)ccc3N)=O)C2C1 C1(CCCSCCNC(=O)Cn2ccnn2)CCCN1C(=O)CCCC1CCC1 N1(C(C=C(C)Cl)=O)CCN(C(C2CCCC(F)(F)CC2)=O)CC1C C(c1cc(F)cc(F)c1)=CC(=O)NCC1CC(OC)CN1C(C1CC(OC)C1)=O C1(C)(C(=O)NCCOCCNC(C2CC(C)(C)C2)=O)COCC1(F)F C1(C(=O)NC(C2CN(C(c3c(OC)c(Cl)sc3)=O)C2)C)CCCC1C1CC1 Cc1csc2ccc(C(=O)N(C)CCN(C(=O)C(F)=CCCF)C)cc12 C(=O)(C#CC1CCCCO1)N1CC(CNC(c2ccnc(O)c2)=O)C(O)C1 C=CCC(CC=C)C(=O)N1CCC(CNC(=O)C(C2CCCCCC2)O)C(C)C1 CC(CCCCN)NC(=O)C(=O)Nc1cccc(C(c2ccc(O)cc2)=O)c1 C1(NC(=O)CC2CC2(Cl)Cl)C2CN(C(c3[nH]nnc3C3CC3)=O)CC12 C(=O)(CCC(=O)N1CCCC(NC(=O)C(c2cccc(F)c2)C)C1)NC.C1CO1 N1(C(c2nc(C(C)C)sc2)=O)CCC(CCNC(=O)COCC2CCOC2)CC1 CCCCC(C(=O)N1CCC(CNC(=O)CC23COC(C)(C2)C3)C1)ON=C(C)C C1(C(=O)NCCCCN(C)C(C2CC3CC3C2)=O)CCC2CC2CC1 C1(CN(C(c2cnc(C)o2)=O)C)COCCN1C(=O)CC1CNC(=O)C1 N1(C(c2ccc(CCC)[nH]2)=O)CCC(F)(CNC(=O)CN2CCCCC2CC)C1 CC1CCC(n2cc(CC3CN(C(c4ccccc4F)=O)C3)nn2)CC1 CC1(C(=O)NC2CC(C(N3CC4(CSC4)C3)=O)CC2O)CC2CC2C1 C(=O)(C1CCCn2ccnc21)NC(CNC(c1n[nH]c(CC)c1Cl)=O)(C)CC c1(CC)cccc(C(=O)NCC2(C)CCCN2C(=O)Cc2ccncc2Cl)n1 N1(C(c2ccc(C)cc2C)=O)CCC(C2CCN(C(=O)Cc3cscn3)CC2)C1 c1(N(C)C)nc(NC(=O)CCCn2cc(-c3c(F)ccnc3F)nn2)cc(Cl)n1 CC(C)C(F)C(=O)NCC1(C(=O)NCC2CCCCC2)CC=CC1 CCCC(C(=O)NCc1ncsn1)NC(=O)C(C1CCCCN1C)C Cc1c(C(=O)N(CC(C)CNC(c2cccnn2)=O)C)c(C(F)(F)F)nn1C C1(CNC(c2c(C)n[nH]c2)=O)CC12CCN(C(c1csc(C)c1C)=O)CC2 CCN(CCO)N1CCC(OCCO)C1.OCC c1(CC(=O)NC2CC(F)(CNC(=O)C(F)(F)c3cscn3)C2)cnccn1 CC1CC(C)CN1C(=O)C.C(=O)(CCC(F)F)NC(c1ccccc1)=O N1(C(Cc2ncc(C)o2)=O)CCCC(CN(C)C(C2(Cl)CC2(F)F)=O)C1 CC1CC2CN(C(=O)NC(C)Cc3cccc(F)c3)CCN2C1=O c1(C(C(=O)NC(C)C)N(C)CCc2ccc(Cl)cc2Cl)ccc([N+](=O)[O-])cc1 C1(NC(C2(CC#C)CCOC2)=O)CC(C)N(C(c2ncoc2C2CCC2)=O)C1 c1(C(N2CCC(F)(CNC(C=CCCC)=O)C2)=O)cc(Cl)c(Cl)cc1OC c1(C(C(=O)NC)NC(c2ccc(OC(F)F)cc2)=O)ccc(Cl)c(C)c1Cl c1(C(C(=O)NCCN(C(c2c(C)snn2)=O)C2CC2)(C)C)cccc(C#N)c1 C1(C(N2CC(N(C(CC(C)NC(=O)OC(C)(C)C)=O)C)C2)=O)CC(=O)NC(=O)N1 CCC(CC(=O)N1CC(C(C)NC(c2cc(SC)c(C)o2)=O)C1)C1CC1 Cc1cc(NC2CCCC2c2ccc(F)cc2)ccn1 C(=O)(C1c2c[nH]nc2CN1C(c1ncn2c1CCC2)=O)N1CC2CC(C)CC2C1 Cc1ccn2c(C(N3CCCC(CNC(C4CCC4(C)C)=O)CC3)=O)cnc2c1 CCCCC(O)C(C)C(=O)N1CC(O)CC1C(=O)N(CCOC)CC C#Cc1ccc(C(N2CCCC(NC(c3cc(CCC)c[nH]3)=O)C2)=O)cc1Cl c1(OC)cccc(C(N2CCC(NC(c3ccnn3C3CC3)=O)C2C2CC2)=O)c1 N1(C(CN(CCOC)C)=O)C(C(=O)Nc2cnc(C#N)nc2)CCC12CC2 N1(C(C2(NC(C)=O)CCCC2)=O)CCC(C)(CNC(=O)C(F)=C2CCC2)C1 c1(NC(c2c(C)oc(C(C)C)n2)=O)ccc2c(c1)CCC(N)C2 C1(NC(=O)Cc2ccccn2)CCN(C(c2cnoc2C2CC2)=O)CC1CO C(=O)(C(O)C(F)F)NCC.c1(N2CC(C)(O)C2=O)cccc(Br)c1.C1CC1 C1(C(N2CCC(C(=O)NC(CNC(=O)OC)C)C2)=O)C2CCC(C2)C1C C1(NC(c2c(C(C)=O)n[nH]c2)=O)CCN(C(=O)CNc2ccc(Cl)cc2)CC1C C1(C(=O)NCC=CC)CCCC1NC(=O)COC1CC=CC1 C(=O)(CCC(C)(C)F)N1CCC(OCC)(OC)C1.C12CCC1(OC)NC2=O C(=O)(C(C)CS(C)=O)NCCC(CNC(C(C=C)(C)C)=O)(C)C O=C(C1CCc2nccn21)NC1CCCC1NC(c1cccc(C(F)F)c1F)=O c1(C(N2CCCC(C)(C)C2)C(=O)NCCCSC)cc(S(N)(=O)=O)cs1 Cc1ccc(F)cc1C(N1CCC(N(C(=O)CCc2cnn[nH]2)C)C(C)C1)=O C(c1ccc(Cl)s1)=CC(=O)N(C)CC1CCCN1C(=O)CSc1nc[nH]n1 n1(CC)ncc(=NC(=O)C2(C)CCC(c3ccccn3)O2)[nH]1 C1(CCNC2CC2)(SC)CCC1.C12(CC1)C(=O)NCCSCC(=O)N2 C=CCC(C(=O)NCc1ncn(C2CC2)n1)NC(c1c[nH]nc1COC)=O c1(C(=O)NC(c2ccns2)C)csc(CNC(=O)C(F)C2CCOC2)c1 C1(CC)CN(C(c2cnn(CCOC)c2)=O)CCC1NC(=O)Cc1sc(C)nc1C n1(CCC(=O)N(CC)CC2CCC(OC)CC2)cc(N)c(O)nc1=O N1(C(c2n[nH]c(CC)c2Cl)=O)CCCC(NC(c2sccc2CO)=O)C1C C(=O)(C(C(C)C)N(C)C(C1CC(C)(O)C1)=O)N1CCC(CNC(=O)OCC)C1 Cc1nnc2n1CCC(C(N1CC3CCC(C1)N3C(=O)C(C)(C)C1CCC1)=O)C2 c1(C(N2CC3C(CNC(c4cccnc4S)=O)C3C2)=O)cc(F)c2[nH]nnc2c1 C(=O)(C(C)CC(C)(C)C)N(C(C)CN(C(=O)C=Cc1cnn(C)c1)C)C C=CC(C)(CCOC)C(=O)N1CCN(C(c2ccc(CC3CC3)s2)=O)CC(C)C1 C1(C(=O)NCC(=O)NCC(CC)C)CSCCN1C(=O)OC(C)(C)C C12(CNC(c3cc(CC)on3)=O)CCC1CN(C(=O)CC1(OC)CCCCC1)C2 C(=O)(CC(O)CC(C)(C)C)N(C(CC)CC(=O)NCc1oc(C)nc1C)C CCCCCC(F)C(=O)NC1(CC(=O)NC2CCCCC2C)CC1 C(=O)(C1c2ccccc2C2CC1C2)N1CC(NC(=O)CC(F)(F)C(F)(F)F)C1 C(=O)(C(C(=O)N1CCC(NC(=O)C=CSC)C1)C(C)(C)C)OCC [N-]=[N+]=NC1CC2(C1)CN(C(C1CCN(C(c3cncc(O)c3)=O)CC1)=O)C2 C(=O)(CC(C)(C)C(F)F)NC1C(CC(=O)NCc2cc(C)on2)CCCC1 C1(C)(NC(C)=O)CCN(C(=O)CC(C2CC2)NC(=O)Cn2cncn2)C1 c1(OC)ccc(C(C)C(N2CC3CC2C3CNC(=O)C(F)(F)C2CC2)=O)cc1 C1(NC(=O)C2CC2)CC2CC(C1)CN(C(c1ccc(-c3ccccc3)cn1)=O)C2 C1(CF)CC(N=c2nc(N3CC(c4nccs4)C3)c3c(Cl)cccc3[nH]2)C1 C(=O)(CC(C)C(C)(C)C)N1CC(NC(c2nnn(CC)c2C)=O)C2(C1)CC2 c1(NC(C(=O)NC(C2CCOC2)C)=O)ccc(OCCOCC(F)(F)F)c(F)c1 C12(C(=O)NCC(CNC(C(CC)NC(N)=O)=O)O)CCCCC(F)(C1)C2 Cc1c(CNC2CCC(C(=O)N(C)CC3(C)COC3)CC2)cnn1C n1(CC=C)nnnc1C(c1cc(OC)ns1)NCCc1ncnn1CCC CCCCC(C(=O)NC1CC1NC(c1cnc(Br)c(O)c1)=O)N(C)C C=CC1(CNC(=O)NC(C(=O)O)C2(O)CCC2)CCCCC1 CC1=NNC(=O)C1CC(N1CCCC1C(C)(C)C(=O)N(C)CC1(CO)CC1)=O Cn1ccnc(NC2CC(CNC(=O)CC3CC4CC4C3)C2)c1=O CC1c2ccc(Cl)cc2CCN1C(c1coc(C2CCCCC2)n1)=O Cc1cnc(NCC2(C)CCCN(C(=O)CCCn3ccccc3=O)C2)nc1O N1(C(c2nc(CC)sc2)=O)CCCC(CCNC(=O)C(O)CC2CCOCC2)C1 Cc1cccnc1C=CC(N1CC2CC1C2CNC(c1ccnn1CCF)=O)=O c1(C(N2CC(NC(C(C)(C)OC)=O)C(C(F)F)C2)=O)cc(=O)c2ccncc2o1 N1(C(C(N2CC(C)C2)C)=O)CCC(NC(C2CC(OC(F)F)C2)=O)C1 N1(Cc2n(C)cnn2)C2CCC1CN(C(c1cc3n(n1)CCCO3)=O)C2 C1(NC(c2cccc(F)c2O)=O)CC2CCC(C1)N2C(C1CC(O)C1)=O N1(C(C(C)N2CCC2)=O)CCC(CN(C)C(=O)CN(c2ccncc2)C)C1 C1(NC(C(COCC=C)c2ccccc2)=O)CCN(c2nc(C)ns2)CC1O C12(C(=O)NC3C4(CN(C(CCCCC=C)=O)C4)SCC3)CCCC(=O)N1CCC2 N1(C(c2nc(C(C)NC(C(CC)C#N)=O)oc2)=O)CC2CCOC(=O)C2C1 C(=O)(C(CC)C(C)O)NC(CCNC(CC1(C=C)CCC1)=O)Cc1ccccc1 C(=O)(CC1=CCCCC1)N(C(C)CNC(=O)CC1COCC(C)(C)O1)C C=CCC(CC(C)C)C(=O)N1CC2CC2(NC(C2CC(=O)N(C(C)C)C2)=O)C1 c1(C(C(=O)NC(C)CN(C(=O)CCSC(F)(F)F)C)OC)ccccc1 CCCCC(O)C(C)C(=O)NCC(C)(C)NC(=O)CS(N)(=O)=O N1(C(C2C(CCC)C2)=O)CCCC(CNC(=O)CC2CC(C)(C)CCO2)CC1 C(=O)(C#CC1CCCCC1)N1C(C)CCC(NC(=O)C=CC2CCOC2)C1 C1(CNC(C(C)OCCC(C)C)=O)CCC(NC(=O)C(C)(C)c2cccnc2)C1 C1(NC(c2onc(C)c2C)=O)(CNC(=O)CCCN(C)C)CCCCC1C C1(C(=O)NCC(CCCC)NC(c2ncoc2C2CCC2)=O)CCOC(=O)CC1 C1(C(N(C2CCN(C(c3ccsc3Cl)=O)C2)CC)=O)CCN(C)C1=O C(=O)(CCC#Cc1ccccc1)N1CCN(C(Cc2c(C)nn(C)c2)=O)C2C1C2 c1(OC)ccc2nc(N3CC(F)(F)CC3CNC(C3CCC4CC4C3)=O)sc2n1 c1(CN(c2ccc(NC(=O)OC(C)(C)C)nc2)C=O)ccc2cccnc2c1 N1(C(C(C)OC)=O)CCCC(C)(C)C1CNC(c1cccn2cncc12)=O C1(C(C)C)CN(C(c2ncnn2C)C(=O)Nc2ccc(Br)cc2)CCO1 Cc1ccc(CC(=O)NCC2COCC2NC(=O)C=CCOC2CCOCC2)cc1 C1(F)(C(=O)NC(C#C)(C)C2CC2)CCCN(C(=O)Cn2nccn2)C1 c1(CN(C)CC2CCN(C(C=CCOCCOC)=O)C2)ccc2ccsc2c1 C(=O)(C#CC1CCCCC1)NCC1CCCCN1CCC(=C)C CC1CC(NC(=O)CC2(C3CC3)CC2)CCN1C(=O)Cn1cccc1 CC1C(NC(c2cnn(CC3CCC3)c2)=O)CC2CCC1N2C(C1(O)COC1)=O C(CNC(c1ncccc1F)=O)(C(C)C(C)C)NC(c1c(C)ncnc1)=O C1(C(=O)NCC(C(=O)NC(CC(CC)C)C)OC)CC2(CC(=O)C2)C1 C1(C(N2CC(CNC(=O)C(C)C)C2)=O)(OC)CN(C(c2ccccc2)=O)C1 N1(C(C(CC)C)=O)CC(C2CCN(C(C3C(C(=O)OC)C3C)=O)CC2)C1 C1(C(=O)NC(c2nc(C(=O)NC3C=CCC3)co2)C)CC12CCCCC2 S(=O)(=O)(c1cccs1)N(CC(=O)NC1CCC(NC(=O)Cc2nc[nH]n2)CC1)C c1(C(=O)NCC2CCCN(C(CCOCCC)=O)C2)c(Cl)oc2ccccc12 C1(C(C)NC(c2cnc(C)[nH]2)=O)CCCN(C(c2csc(C3CC3)n2)=O)C1 CCC(C)(C)C(O)C(=O)NC1CC(CNC(c2occ3c2CCC3)=O)C1 N1(C(C(CCSC)O)=O)CC2CC(NC(=O)CCC3CC(F)(F)C3)CC1C2 C1(C)(CC(=O)NC(CCC=C)C)CCN(C(c2cnc(CC)o2)=O)C1 C12(NC(c3n[nH]c(CC)c3Cl)=O)COCCC1CN(C(=O)C(C)(C)SC)C2 C1(C(=O)NCCCCCC=C)N(C(=O)C(F)CCC)CCCC1(C)C O=C(CCS(=O)(=O)Cc1ccccc1)NC1CC(F)(CNC(c2cnc[nH]2)=O)C1 C1(C(=O)NC(C)CCCCNC(c2cc(C#N)c[nH]2)=O)CC12CC(F)(F)C2 C(=O)(CC1=CCCCC1)N1C(CC)C(C(=O)NC(C)C(C)(C)C)CC1 N1(C(=O)COC(F)F)CCCCC(NC(C2C3CCC2(c2cncs2)C3)=O)C1 N1(C(C(CC)C)=O)CCC(C)(NC(c2cc(N(C)C)ccn2)=O)CC1 Cc1scc(C(=O)NCC(C)N(C(=O)C=CC(C)C)C)c1C c1(-c2cn(CCC(N3CCCC(COC)C3)=O)nn2)c(C)cccc1C CCC(F)(F)C(C)(C)C(=O)NCC1(C)CCCN(C(=O)CCn2ccnc2C)C1 c1(C(=O)NC(CNC(C(C=C)(C)CC)=O)(C)C2CCC2)cc(F)c(F)c(C#N)c1 c1(Nc2cc(N3CCN(C)C(C(F)(F)F)C3)ncn2)cc2nc[nH]c2cn1 C(=O)(C(CO)C(C)(C)C)N1CC2C(NC(c3nc(C(C)C)oc3)=O)C2C1 C#CC1(C(N2CCC(c3nc(N(C)C)no3)(C(=O)OC)C2)=O)CCNC1 C1(CNC(C2N(CC)CCC2)=O)CN(C(=O)CCCSC)CC(C)(C)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(O)CC1C(=O)NC(C)(C)C#CC c1(C(=O)NC2CC(CCNC(c3cccc(C)n3)=O)C2)cc2c(nn1)OCCS2 c1(CNCC2N(C(C3CC(=O)NC3)=O)CCOC2)c[nH]c2cc(Cl)ccc12 C(C(CC(C)C)C(=O)OC)OCCCN(CCCC)C Cc1c[nH]nc1C(C1(C(=O)NC(n2cc(CCN(C)C)nn2)C2CC2)CC1)(F)F.C1CC1 C1(NC(COC2(C)CCC2)=O)CN(C(c2cc(C3CC3)n(C(F)F)n2)=O)CC1F N1(C(C(C)n2cccc2)=O)CCC(NC(C2CC2(F)F)=O)C1C C1(C(=O)NCCC2CCC(C)(C)O2)CN(C(C2(CO)CCC2)=O)CC12CC2 CC(CC1CCC1)CCC(=O)NC1CCCC(c2ccccc2)C1 C1(NC(=O)CCC2CC2(Cl)Cl)CCC(NC(C2(C(N)=O)CC2)=O)CC1 C1(n2c(-c3c(CCC)n[nH]c3)nc(-c3nccs3)n2)CC12CCc1ccccc12 c1(NC(CNC(c2c(OC)cc(F)cc2)=O)CO)ncnc2scc(Br)c12 Cc1cc(C(=O)NCCNCc2ccc3nc[nH]c3c2)cc(C)c1F C(=O)(N=c1nc2ccccn2[nH]1)N1CC(C)N(c2ccc(F)c(F)c2)CC1 O=C1OC2CC1N(C(C1(F)CCN(C(c3cncc(F)c3)=O)C1)=O)C2 c1(C(N2CCC(NC(CCCOCC)=O)CC2)=O)cn(C)c(=O)c(C)n1 c1(NC(N2C(C(N3CCC(C)CC3)=O)CCC2)=O)cncc([N+](=O)[O-])c1 c1(OC)cccc2c1OC(C(=O)NC1(C)CN(C(=O)C=Cc3cnn(C)c3)C1)C2 C1(NC(CN(CCOC)C)=O)CN(C(=O)C=C(C)c2cccs2)CC1(C)C c1(C(=O)NC(CNC(c2cc(C)nc(O)c2)=O)C2CCC2)ccc2c(n1)NCC2 c1(C(=O)NCCOCCN(C)C(C2CCO2)=O)cccc(CC2CC2)c1 N1(C(CCC(=C)Cl)=O)CCN(C(c2cc3sc(CC)cc3s2)=O)C(C)CC1C CC1(C)COCC1C(=O)NC(C1CCN(C(=O)Cc2ccc(F)cn2)CC1)CO C1(C(N2CCC(N(C(C=CCC)=O)CC)C2)=O)CCCCCC1(F)F C1(O)(CC)CCCN(C(=O)C(CNC(=O)CCc2ccccc2)OC(C)C)C1 N1(C(c2cnn(C)c2)C(=O)NC(C)C)CC(C2(O)CCC2)C12CCC2 O=C(C1=CCN(C(=O)C(Cl)Cl)C1)NC1CCOCC1F CCC(CC)C(C(=O)N1CCN(C(=O)CCS(C)=O)CC1)N1CCOCC1 C1(CN(C(C)C(=O)NC(C)(C)C)C)CCN(C(=O)CC2CCCC2O)CC1 C1(N(C(=O)CCCC(N)=O)C23C(CN(C(CC4(C)CC4)=O)C2)C3)CNC(=O)C(C)(C)C1 C(=O)(C1=CCN(C(=O)CCc2cnn(C)c2)CC1)NC1C(CC)CCCC1 c1(C(C(=O)NCC(C2CC2)NC(C2(OC)CCCC2)=O)(F)F)ccc(F)cc1F n1(CC)cc(CC(=O)NC(C2CN(C(=O)C(C)C3CCCO3)C2)C)cn1 c1(C(=O)NCCN(C(c2ncc(C)cc2C)=O)C2CC2)cnc2scnc2c1 N1(C(c2c(C)c[nH]n2)=O)CCOC(CNC(=O)C(C)(C)Cc2cccc(Cl)c2)C1 CN1CC(O)CCC1C(=O)NCC1CCCC1C(=O)NCCSCCO C1(COC)CN(C(=O)C(N2CCC(C)C2)=O)CCN1C(=O)CC1CC(F)(F)C1 CC1CCN(C(=O)C=CC(C)(C)NC(C2CCOC2)=O)CCS1 C(=O)(C1=NOC2(CCC2)C1)NC1CCC(NC(c2ccc(SCC)nc2)=O)CC1 c1(CNCCCC2N(C)CCCC2)cccc(Br)c1F C1(CNC(NCc2c(C)c(Cl)ccc2)=S)CCS(=O)(=O)C(C)C1 N1(C(=O)CCCc2cncc(Br)c2)CCCC(n2cc(C3(O)CSC3)nn2)C1 C1(N(C(=O)CCC2CCCOC2)C)CCC(NC(=O)CCN2CCC(F)C2)CC1 C1(C(N2CCCC(C)(NC(c3n[nH]c4c3CCC4)=O)C2)=O)CCOCC12CCC2 C(CS(=O)(=O)CC(=O)N1CCC(C)(CNC(=O)CC2CC3CCC2C3)C1)OC C1(NC(C(CNC(COCCSC)=O)CC2CC2)=O)CC(C)OC(C)C1 Cc1ccc(C=CC(N2C(C(=O)N(C3CCC3)CC(C)C)CCC2CO)=O)cc1 c1(NC(C2N(C(c3c(C)noc3C)=O)CCNC2)=O)cc(Br)cnc1C(N)=O C(=O)(C1CCCc2ncccc21)NC(CN(C(C(CCCC)C)=O)C)C c1(C(=O)NCCC(C)N(C(=O)CS(N)(=O)=O)C)sc2cc(F)ccc2c1Cl CC1(C)CC(O)(CC(N2CCOC(CNC(=O)CCN3CCOCC3)C2)=O)CO1 C1(CNC(C2C(=C)C2)=O)CC(F)(CNC(=O)CNC(=O)Nc2ccsc2)C1 C(=O)(CCCCCC#N)NC1(C(=O)NCC(CC)(C)C)CC(CO)C1 C12N(CCC1(C)C)C(=O)C(C)C(=O)C(CC(C#C)C)CN(C)C2=O CCC(C)CC(CCO)N(Cc1cscc1Br)Cc1ccc(SC)cc1 C1(C(N(CCCCN(C(c2cc(C)c(=N)[nH]c2)=O)C)C)=O)CCn2cnnc2C1 C1(C)(C(=O)NC(c2cccnc2)C(=O)N(CC(C(=O)OC)C)C)CNC(=O)C1 Cn1ccc(=NC(=O)C2CN(C(C3CC(C4CC4)=NO3)=O)CC2(F)F)[nH]1 N1(C(c2c(C)ccc(CC)c2)=O)CCCC1C1CCCN1C(c1cccn1C)=O Cc1csc(CC(=O)NC2CC(NC(=O)CCOCC(F)F)C2)n1 CCC(CSC)CC(=O)NCCCC(c1ccccc1)NC(c1ccc(O)nc1)=O c1(C(=O)NCC(CNC(C(C)N(C(C)=O)C)=O)CO)cnn2cc(C#N)cnc12 N(C)(S(=O)(=O)N(C)C)CC(=O)NC(CC)(CNC(=O)C(C)n1cccn1)CC c1(C(=O)NC2(C)CN(C(c3c(C)con3)=O)C2)ccn(CCO)c1C CCC(COC)(CC)C(=O)NC1CCN(C(=O)Cn2nc(O)ccc2=O)CC1C NS(=O)(=O)C1(C(=O)NCC2CC(NC(C3(CF)CC3)=O)CC2O)CCCC1 c1(C2CCN(C(C(=O)NCCCC)c3cc[nH]n3)C2C)ccc(C)c(C)c1 C1(CNC(=O)Nc2cc(CC)ncn2)C2C=CC(C2)N1C(=O)OC(C)(C)C O=S(=O)(c1cccc(=NCC(F)c2ccccc2)[nH]1)N1CCC(SC(F)F)C1 c1(C(C)(F)F)nc(C(=O)NCc2cn(CCNC(=O)CC(=O)N(C)C)nn2)cs1 c1(C(=O)NC(CCCNC(CCCOC)=O)(C)C)cc(Cl)c2n[nH]cc2c1 c1(C(N2C(CN(C)C(C3CC3C(C)(F)F)=O)CCC2)=O)cccc2sccc12 C1(C(N2CCC(C(CO)NC(C3(C#C)CCCC3)=O)CC2)=O)CCOCC1(C)C CCCCCC(C)CC(=O)NC1CC(C(=O)N(C(C)CC)CC)C12CCC2 CC1=NOC(C)(C(=O)NCC2CN(C(=O)CCN3C(=O)CCC3=O)CCO2)C1 Cc1noc2ncnc(NC3CC(NC(=O)CCC(C)(C)F)C3)c12 c1(COC(=O)Nc2ccc(CC)cc2)cc(F)cc2c1OCOC2.C(=O)CC N1(C(Cn2nc(C)c(Cl)c2C)=O)CCN(C(C2CC2C2CCC2)=O)CCC1C Cc1ccc(C(=O)NCC(O)CNC(c2ccc(Cn3ccnn3)o2)=O)o1 C1(NC(C=C(C)C)=O)CCC2(CC1)CN(C(=O)N=c1[nH][nH]cc1I)C2 c1(OC)cncc(C(N2CCC(NC(C3(c4ccsc4)CC3)=O)C(O)C2)=O)c1C Cc1nc(=N)[nH]cc1C(=O)NCC1CCC1NC(c1ccnn(C)c1=O)=O c1(C(=O)NCC(C2CCCCC2)(C)NC(C)=O)ccc2nccn2c1 Cc1cnccc1C(=O)NCCN1CCN(C(C2(C)CC2C)=O)CC1 N1(C(C(c2c(C)nn(C)c2)C)=O)CCCCC(NC(c2ccc(N)c(Cl)n2)=O)C1 C1(NC(c2c(CC(=O)OC)cccc2)=O)CCC(C)N(C(c2csnc2C)=O)C1 C(C)(c1ccc(CC)cc1)=CC(N1CC(CNC(C=CC=CC)=O)C(C)C1)=O c1(N2CCC(C(C)O)C2)ccc(NC(=O)CSCc2ccccc2Cl)cn1 c1(C(CC)C(=O)N(CC(C)NC(=O)Cc2cnoc2)C)ccc(Br)cc1 c1(C(N2CCC(Sc3ccccc3)C2)C(=O)NCC)cccc(COCCF)c1 C1(C(N(C(C)CC2CC2)C)=O)(NC(=O)CCC2CC2(F)F)CCOC1 C1(C2CCN(C(c3ccnc(F)c3O)=O)CC2)(NC(=O)Cc2ccoc2)CCC1 C1(OC)CC2CCC1CC2C(=O)NCC1(F)CC(NC(C2SCCCS2)=O)C1 N1(C(C2(CSC)CC2)=O)CCC(CCC(=O)Nc2ccccc2F)CC1 c1(C(=O)Nc2c(C)cnc(Cl)c2)ccc2c(C(N3CCC(C)(O)C3)=O)n[nH]c2c1 C=CCCN=C(NCC(C)C(F)F)N1CCCCC(S(C)(=O)=O)C1 c1(C(=O)NC2CN(C(c3ccc(CC=C)cc3)=O)C2)cc(Cl)cc(C)c1OC c1(CC)cc2nn(C)cc2cc1Sc1ccc(C(C)(C)C)nc1 N#CC1(NC(C2CC2c2ccccc2)=O)CC2(CCC2)C1 Nc1sc2c(c1C(=O)NCC1CCCC1NC(=O)C(O)CC1CC1)CCC2 C1(NC(CCNC(C)=O)=O)CCSC12CN(C(c1cc(C(C)(C)C)[nH]c1C)=O)C2 c1(C(=O)NCCOCCN(C2COC2)C(c2ccccc2)=O)cc(C(F)(F)F)n[nH]1 c1(CC(C(=O)Nc2n[nH]c(C)c2-c2ccccc2)C)ccc(C#N)cc1 CC(=O)CCN=C(NCC1COC(C)(C)O1)NCC(C)(C)C(N)=O N1(C(CC)=O)C2CCC1CC(NC(c1cc(OC)nc(Cl)c1)=O)C2 N1(C(C(C(=O)OC)OC)=O)CCC(NC(c2c(Cl)sc(C)c2C)=O)C(O)C1 N12CC3(CN(CC3CO)C(=O)c3nc1cc(O)n3)C2.c1(COC)ccn(C)c1 c1(CC(=O)NC2(COCC)CN(C(C3(CF)COC3)=O)C2)ccc(F)cc1F C1(C)(C(N2CC(CCNC(C3CCC3c3nc[nH]n3)=O)(OC)C2)=O)CCNC1=O c1(C(=O)NC(C(C)NC(CSCC(C)C)=O)CO)cc2ccccc2s1 Cc1ccc(C(=O)NC2CCC2NC(=O)COC(C)C)cc1Br N1(C(c2nc(C)c(C#N)cc2)=O)Cc2nccn2CC(NC(=O)CCCF)C1 C(CC(=O)NCc1csc(O)n1)(C(F)F)NC(c1c(C)oc(CO)c1)=O Cc1nc([N+](=O)[O-])cn1CC(=O)N(CC(C)CNC(=O)CN1CCC(C)(O)C1)C c1(OC)ccc(C2C(=O)OCCN2C2CCCO2)cc1.C(=O)(CSCC(F)F)SC C1(CNC(c2cc3n(n2)CCC3)=O)CCC12CCN(C(C1CCOC1)=O)CC2 c1(C(N2C(CCNC(COC(C)C)=O)CCCC2)=O)cccc2c1CCOC2 c1(C(N2CCCC(NC(C(CN(C)C)(F)F)=O)C2)=O)cc(O)ncc1Br C1(OC)CC(NC(=O)CN(C)C(N)=O)CN(C(c2ncnn2C)=O)C1 c1(C(N2CC(NC(=O)C(F)F)CC(OC)C2)=O)ccc2c(c1)C(=O)CCN2 S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1C2(CC(C(=O)OCC)C2)CC1 N1(C(c2cnc(C)n2C)=O)CCN(C(c2cccnc2O)=O)C(C2CC2)C1 C(CCCC(F)(F)C(F)(F)F)NCc1ccc(C(=O)OCC)s1 C1(CNC(Cn2c(C)ccn2)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC1(F)F C(=O)(C1=CC(C)(C)C1)N(C(C)(C)CC(=O)NCC1CCC(C2CC2)O1)C C123CC(C1)(OC2C)CNC3=O.C(C(=O)NC1CC1CF)SCCOC C1(NC(=O)CC2CNC(=O)O2)CCC(NC(C2(CF)CC(F)(F)C2)=O)CC1 CCC(C(=O)N(C)Cc1cccs1)NC(c1ccc(SC)o1)=O N1(C(=O)Nc2ncc(-c3ccc(F)nc3)cn2)C2CCCC1COC2 C1(C(N2CC(F)CC(NC(COCCC(C)C)=O)C2)=O)CCC2(CC1)CC(O)C2 N1(C(c2cnn(C(C)C)c2F)=O)CCC2CCC12CNC(=O)CCC(N)=O Cc1nn2ncccc2c1C(=O)NCC(C1CC1)N(C(=O)C=CC1CC1)C C(=O)(C1=CS(=O)(=O)CCC1)NC1CCC(CN(C(C(CC)SC)=O)C)CC1 CCC(C(=O)NCCN(C1CCCC1)C(c1c[nH]c(=N)s1)=O)Oc1ccccc1 N1(C(CCCCCOCC)=O)CC2(C)CN(C(=O)CN3CCC3)CC2(C)C1 C1(C(N2CCN(C(c3c(OC)n[nH]c3)=O)C(C)C2)=O)COc2cc(F)ccc2C1 C1(C2CCC(NCC(N)CC3CCC(=O)N3C)CC2)(C(C)C)CC1 C12(C(N3CCCC(O)(CCNC(C4CCCC4)=O)C3)=O)CC1Cc1c[nH]nc12 N1(C(=O)CNC(=O)OC)CC2CC(NC(c3c(CC)noc3)=O)C2C1 C1(C)(C(=O)NCc2c(C(=O)NC(C)(C(C)OC)C3CC3)nco2)CCOCC1 c1(C(=O)NCCC2(O)CN(C(C(C)NC(COC)=O)=O)C2)c(C)cccc1Cl c1(OC)ccc2cc(C(=O)NC3CCC3NC(c3cnc(C)s3)=O)ccc2c1 c1(OC)cc(CC(N2CC(CCNC(C3(C)C=CCC3)=O)C2)=O)cc(F)c1 CN1CCOCC1C(N1CC(CNC(C2(N3CCCCC3=O)CC2)=O)C1)=O C(C1CCN(C(c2ccccc2Cl)=O)CC1)=CC(=O)N(C)CCN1CCCCC1 N1(C(CSc2cn(C)nc2)=O)CCN(C(C2CCC3CC3CC2)=O)CC1CF C1(CNC(C2CC(C#C)(O)C2)=O)C(C2CC2)CCN1C(c1ccc(C)cc1)=O c1(CCC)nnc(S)n1CC(=O)NC(C)CCNC(c1ccn(C)n1)=O c1(N2CCC(CCNC(C3(C)CC=CCC3)=O)CC2)ncnn2cccc12 C1(O)(CC(=O)NC2C(CCC)C2)CCCOC1.C12(CC1)C(=O)N2.C1(C)CC1 c1(C(N2CCC(O)(C(C)NC(=O)Cc3cncnc3)C2)=O)cc(Cl)c(Cl)cc1N C1(C(=O)NCCCCC)CC(F)CN(Cc2nn(C)cc2Br)C1 N1(C(c2csc3ccc(Br)cc23)C(=O)NCC=C)CCn2c(C)nnc2C1 Cc1ncnc(C)c1C1(NC(=O)CC(C)(C)CN(C(=O)C=CBr)C)CC1 N1(C(C2C(OC)CCCC2)=O)CCC(C)N(C(c2csnc2C)=O)CC1 c1(CNC2(CCO)CCCC2)cc2cncc(Br)c2o1 N=c1[nH]cncc1C(=O)NC1CC(CNC(=O)CC2CSCCS2)C1 C(C1CCCCCC1)=CC(=O)NC1(C)CN(C(C(C)c2cccs2)=O)C1 C=CCCCCCCCC(=O)N1CCN(C(=O)C=Cc2cocn2)C(C)C1C C1(NC(=O)COCCOCCO)CC(O)CN1C=O.c1(O)cnn(CC(F)(F)F)c1 CN1CCN(C(=O)CC2CCN2C(=O)COC(C)(C)C)CC(O)C1 N1(C(C2=CC(C)(CC)C2)=O)CCC2(CCOCC2)C(NC(C2(COC)CC2)=O)C1 N1(C(C)C)C(=O)COCC1C(=O)NC1CCCN(C(=O)CNc2ccccc2)C1 CC(CC(C)(F)F)C(=O)N1CC(NC(c2cc3c([nH]2)CCCC3)=O)C(C(F)F)C1 c1(CC)nc(C)[nH]c1C(=O)NC1CC12CC(NC(=O)CCc1cnoc1)C2 N1(C(C2C3CN(C(c4cc(OC)c(I)cc4)=O)CC32)=O)CCOC2(CCOC2)C1 C(=O)(CP(C)(C)=O)N(C1CCC(NC(=O)CCCN2CCCC2)CC1)C C(=O)(C1Cc2ccc(Cl)cc21)NC1(CNC(C=CC(N)=O)=O)CCCCC1 CC(CC(=O)N(C(CNC(=O)COCC1CC1)C1CC1)C)c1cccnc1 c1(C(=O)NC2C(NC(C(C)NC(c3ccco3)=O)=O)C2)c(Cl)ccc(Br)c1F Cc1ccc(SCC(N2CCCC2C(C)NC(c2cnc(Cl)[nH]2)=O)=O)cc1C CC1(C)CC(NC(=O)CCC23CCC(CC2)C3)CN1C(c1ccc(C#N)cc1)=O CCCC(C1CC1)NC(C1CCC1CNC(=O)C=C(C)C(F)F)=O c1(CC(=O)NCC2CN(C(CCN(C)CCO)=O)C2)c(Cl)ccc(O)c1Cl N1(C(C(C=C)O)=O)CC2CCC(C1)N2C(=O)COCc1nc2ccccc2s1 C1(CC)CCN(C(=O)Cn2cc(CO)nn2)C(C(=O)N2CCCCS2)C1 c1(C(=O)NCC(C)NC(c2ncc(C3CC3)cc2F)=O)c(Cl)ccc(O)c1N Cc1cc(Br)c(NC(C2CC3CC3N2C(c2nc[nH]n2)=O)=O)cc1C N1(C(C2CCC(=O)OCC2)=O)CCC2(CCC(NC(C3CCSC3)=O)C2)CC1 CC(C)CC(C(=O)N1CC(OCCNC(C2CCNC2=O)=O)C1)C(C)C C1(C(N2C3C(NC(CC(CC)C)=O)C(C3)C2)=O)CC(S(C)(=O)=O)C1 C12(C(N3C(CCC(C)(C)NC(C)=O)CCCC3)=O)CC(C)(C1)OC2C c1(C(=O)NC(CC(C)NC(C2CC(=O)C2(C)C)=O)C)ncn2ccccc12 c1(N2CC(CC)SCC2)nc(=NCc2cccc(OC)n2)[nH]c2c1COC2 C(c1ccc(C(N)=O)o1)=CC(=O)NCC1C(CNC(C=C(C)C(C)C)=O)C1 c1(OC)cnccc1CN1CCCCC1CCNC(C1(F)CCC1)=O c1(C2CCN(C(c3c(C(=O)OC)csc3)=O)C2)cccc(F)c1 N1(C(CS(CC(C)C)(=O)=O)=O)CC(NC(=O)CC2CC2)C2(CCS(=O)(=O)CC2)C1 Cc1cc(=NCC(c2cnn(C)c2)N2CCOCC2)[nH]c(C(C)O)n1 C(=O)(C1Cc2ccc(Cl)cc21)NCC(=O)NCC1CCC2(CC1)CC2C1CC1 N1(C(C(c2c(C)cno2)=O)=O)CC(C(C)(C)C)CC(COC(C)(C)C)C1 N1(C(C2(CCOC)CC2)=O)CC2CC2(CNC(C2(C)CC(F)(F)C2)=O)C1 C1(C(=O)NCC(C(CC)CC)O)N(C(=O)CCOC)CC12CCCC2 C1(C(=O)NC(COC)C(C)C)CNC(=O)CC12CCOC2 C(CC#CC)(C(=O)NC(CC)CCO)NC(C1(CC#C)CCOC1)=O c1(C(=O)NCC(CC)NC(=O)CCCC2CCC2)cccc2nc(C(C)C)[nH]c12 N1(c2ccnc(SC)n2)CC2(C1)C(CNC(=O)C1=CCCOCC1)CCS2(=O)=O Cc1nc(NC23CCC(CC2NC(c2nn(C)cc2Cl)=O)C3)ccc1C#N C1C(O)CC(=O)N2CCCC2c2cn1nn2.Cc1cnc(CC(=O)N(C)C)s1 C1(C(=O)OC(C(CCC=C)(C)O)=O)(NC(C(C)OCC#C)=O)CCCCC1 C1(C(N2CCC(C(C)NC(CCOC(C)C)=O)CC2)=O)CCN(C)C(C)C1 N1(C(c2cc(COC)on2)=O)CCCN(C(C23CC(OC)(C2)C3)=O)C(C)C1 C(=O)(C1=CCCN(C(=O)C(O)CC(F)(F)F)C1)NCc1ccn(C)c1 c1(C(=O)NCCC(C)N(C(=O)Cc2cccs2)C)cc(Cl)ccc1[N+](=O)[O-] c1(CC(C)NC(C23CC2CNC3=O)=O)cccc(F)c1 C1(OCC)CC(CNC(=O)CN(C(=O)C(C)=CC(C)(C)C)C)C1 C1(NC(c2[nH]cc(N(C)C)c2)=O)CC(C(=O)N2CC(CC3CCC3)C2)=CC1O c1(C(=O)NC2(CNC(c3ccc(C(C)(C)C)o3)=O)CCC2)ccc2c(n1)CCC2 N1(C(C)C)CCC(C(=O)NCC23CC2CN(C(=O)C2=CCOC2)C3)CC1 N#Cc1cc2occc2c(=O)n1NC(=O)Cc1ccc(Br)c(F)c1 N1(C(C(C(C(C)C)O)(F)F)=O)CCC2(CCCN(C(=O)Cc3cccn3C)C2)C1 c1(C(N(CCNC(=O)C2=CCCC2)CC)=O)cccc2sccc12 c1(CN2CC3(C(C(=O)NC(COC)COC)C3)C2)c(OC(F)(F)F)cccc1F Cc1cncc(C(N2CCCC2(C)C(=O)NC2C=CC(C(=O)N(C)C)C2)=O)n1 C1(COC)C(C)CCCN1N(Cc1cncs1)Cc1ccccc1F N1(C(c2cc(C)sc2)=O)CCC(NC(C2CC2C)=O)CC1 C#CC1CCCC(CNC(=O)CC2C3CCC(C3)N2C(=O)CC(C)(C)C2CC2)C1 C(CCCCNC(=O)CC1(C)CC1(Cl)Cl)NC(C=CCOC)=O C=C(C)CC(C)C(=O)N1CCOCC1CNC(c1ccc(-c2ncon2)cc1)=O N1(c2nnc(-c3cc(=NC)[nH]cc3)n2CCC(C)C)CCOC2(CCSC2)C1 Cc1nc(C(N2CC=CC(NC(=O)CCNC(N)=O)C2)=O)nn1C c1(N(C(c2nccs2)C)C)nccc(=NC2CCC(F)(F)C2)[nH]1 CCC(C)(C)C(C)CC(=O)NCCOCCNC(c1ccc2snnc2c1)=O c1(CC=C(C)C)cc(C(=O)NCC(=C2CN(C(C3CC3F)=O)C2)F)ccc1F C#CCCC(O)C(=O)N1CCCC(CNC(c2conc2COC)=O)C1 c1(NC(C)=O)ccc(Br)cc1C(=O)NCC1CC1NC(c1ccnnc1C)=O CCCC(C)C(=O)NC(C)C(C)NC(c1csc(C)n1)=O C12(C(C)Nc3c(N(C)C(N)=O)cccn3)CCC(CC1)CC2 n1(SCC)ncc(-c2cn(C3CN(C(=O)Cc4csc(C5CC5)n4)C3)nn2)c1C C1(NC(c2cccc(SCC)c2)=O)CC2CC(C1)N(C(c1ccn(C)n1)=O)C2 C(=O)(CCCCC(F)(F)F)N1CC(NC(C(C)OC)=O)C2(C1)CC2 N1(C(C(COC)C)=O)CCC(C2CCN(C(=O)Cc3c(C)nn(C)c3C)CC2)C1 N1(C(COc2ccc(OC)c(C)c2)=O)CC2CCC(C1)N2C(=O)C1=CCCOC1 C1(C(COC)NC(=O)CC2(O)CCCC2)CCCCN1C(=O)C1CC1 c1(C(=O)NCCC2CC(C(=O)NCCc3cc(CC)no3)C2)ncc(F)cn1 Cn1ccn2ncc(C(N3CCC(NC(c4scnc4Cl)=O)C(CO)CC3)=O)c12 Cc1ccc(C(N2CCCC(n3ccnn3)CC2)C(=O)NCCC#N)c(F)c1F Cc1cccc(O)c1C(=O)NC(C)C=CC(=O)NCC(c1cccs1)C c1(C(N2CCCC(N(C(C(CC#C)C)=O)C)CC2)=O)cc([N+](=O)[O-])c(C)cc1C Cc1csc2ncnc(N3CCC(NC(=O)C(C)CC(C)C)C(F)C3)c12 C(=O)(C(CC(F)F)N(C)C(c1cc(C#N)n(C)n1)=O)NC(c1nc(CC)[nH]n1)C C1(C(CNC(CCCN(C)C)=O)(C)O)CCCN(C(=O)CN2CCCS2(=O)=O)C1 c1(C(=O)NCC(CC)(CC)NC(c2cnsc2)=O)cc(NC2CC2)ncc1Cl C1(N(CCN(C(c2nc(C)c(C(C)(C)C)s2)=O)C(C)C)C)CN(CC)CC1(C)C C1(c2n(-c3ccccc3)nnn2)(NC2C3CCCC23)CC2COCC2C1 C1(C(N2CC(CCNC(C3C=C(C)CS3)=O)OCC2)=O)CCCC1C1CC1 C1(NC(c2c(C)[nH]nc2Cl)=O)CN(C(C2CCCCN2C(N)=O)=O)CC2(CC2)C1 C1(CNC(CC2C(C)=NOC2=O)=O)CN(C)CCN1C(=O)C=CC1CC1 C(N=c1[nH]c(C(F)F)nc(=N)[nH]1)c1cc(C(N(CCC(N)=O)C)=O)no1 N1(CCCCNC(C(CN(C)C)O)=O)CCN(C(=O)CC2(O)CCC2)CC1 CC(F)(F)C(C)(C)C(=O)NC1CCN(C(c2cc(N)ccn2)=O)C2CC12 c1(OC)ccc(I)cc1NC(C1CN(C(c2ocnc2C)=O)CCC1O)=O C1(C(C)C)OCCC1C(=O)NCCn1cc(C(=O)N(CC(O)C2CC2)C)cn1 c1(C(N(CCn2cc(CCC#N)nn2)CC)=O)ccc(P(C)(C)=O)o1 C1(C(=O)NCCC2C(C)CCCN2C(=O)COCCF)CN2CCCN1CC2 C(=O)(C(CC)(CC)CC)N1CCC(O)(CNC(CCCCC=C)=O)CC1 C1(C(N2CC(C)(CSC)C2)=O)(CC)CCCN(C(c2ccncc2N)=O)C1 N1(C(c2ccccc2I)C(=O)NC)CCC(O)(c2ccc(C#N)cc2)CC1 N1(C(c2coc(O)n2)=O)CC(CNC(C2(c3ccccc3F)CC2)=O)C2(CC2)C1 C(=O)(CCP(C)(C)=O)N1C(C2(C(N3CC(C)C(F)C3)=O)CC2)CCCC1 C1(C)(C(N(CCN(C(C(CC)COC)=O)C(C)C)C)=O)CCC(F)(F)C1 C1(NC(c2ccc(CSCn3cc(C4C(C)C4)nn3)cc2)=O)CN(C)CC(C)O1 c1(OC)ccc(C(=O)NCCC(O)CNC(C2CCCN2C)=O)c(N)c1F c1(C(C)NC(c2nc(CCOC)oc2)=O)ccc(CNC(C2CC2(F)F)=O)cc1 C(C(CC(C)C)NC(=O)Cn1nc(C)oc1=O)NC(c1c(C)ocn1)=O c1(C(=O)NCC(C)NC(c2c(C)oc(Cl)n2)=O)noc2c1CCCC2 C1(CNC(c2ccccc2F)=O)CN(C(c2cc(Cl)cnn2)=O)C2CC12 C1(F)(C(N2C(CO)CC(C)C2)=O)CS(=O)(=O)CC12CCC2 C1(N(C(C(C=C)O)=O)CC)CCN(C(=O)C(C)(C)Nc2ccccn2)CC1 C(CNCc1cnsc1C)(C(C)C(C)C)NC(c1ncc(C(=O)OCC)s1)=O C1(C(=O)OC)CCC2CN(C(=O)C(Cc3ccccc3)CN)CC2C1 CC1CN(C(c2ccnc(O)c2)=O)CCC1C(=O)NC(C)CCCCO N1(C(C(C)P(C)(C)=O)=O)CCN(C(c2ccco2)=O)CC2CCCCC12 c1(CC(C)NC(C2(CNC(=O)CC3COC(C)C3)CCC2)=O)cnn(C)c1 C1(C)(NC(Cc2c(C)nn(C)c2)=O)CCN(C(c2ccno2)=O)CC1 Cc1ccc(NC(=O)CC23CCC2CN(C(C2CC(CF)C2)=O)C3)c(C)c1 C1(CC(=O)NCCN(CCC)C(C2(C(C)(F)F)CC2)=O)C=CCCC1 CCC(C)CCC(=O)N(CC(O)CNC(c1sc(Br)nc1C)=O)C c1(OC)c(C(N2CCC(C)N(C(C3CC(=O)N(C)C3)=O)CC2)=O)nc(O)nc1O c1(OC)cc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2nnc(O)s2)ccc1Cl c1(CC)noc(CCNC(=O)C(CC)N(C)C(c2ccc(C(C)C)o2)=O)n1 C1(C(=O)NCCC2CCN(C(CCOC(CC(C)C)C)=O)C2)CCOC(=O)CC1 c1(OCC)c(F)cc(C(=O)OC)cc1S(=O)(=O)NCc1cncc2nc(C)[nH]c12 CC1(NC(c2cnnn2C2CCOCC2)=O)CCN(C(c2ncc[nH]c2=O)=O)C1 N1(C(CCSCCCC)=O)CCC(N=c2[nH]nc(C(F)(F)F)s2)(CO)C1 c1(CN(CC(=O)Nc2cccc(-c3ccno3)c2)C)ccc2ccccc2c1O c1(C(N2CCC(N(C(c3c(OC)c(C)ccc3)=O)C)C2)=O)cc(F)cc(Br)c1Cl CC1CN(C(=O)C(n2ccnc2)C2CC2)CC1CNC(=O)C(C)CC#N C1(C(N(C)CC2CCOC2)=O)CN(C(C2CC=CC2)=O)CC(C)(C)C1 c1(C(=O)NCC(N(C(=O)C=C2CCSCC2)C)C2CC2)ccc(F)c(Cl)n1 C1(CNC(c2c(C)nc(O)s2)=O)CCCN(C(=O)C(C)N2CCCC2)CC1 c1(C(=O)NC2CCCN(C(C(CCC)O)=O)C2)cc2ccc(F)cc2nc1O CC(C)(CNC(=O)CC1(CNC(C2CCCC(=O)C2)=O)CC1)CC(F)F S(=O)(=O)(c1ccc(N(C)CCN(C)CCO)cc1Br)NC1C(SC)CCCC1 C1(C(N2CCC=C(F)C2)=O)CCCCCN(C(C2(F)CCC2)=O)C1 c1(SC)cnc(C(c2nnnn2C2CCCC2)NCCc2ccno2)s1 c1(CCCC(=O)NC2CCCC2NC(C2CC2C(F)F)=O)cccc(Cl)c1 C1(NC(C(CC)SC)=O)CCCC(CNC(c2ccc(C3(F)COC3)cc2)=O)C1 C1(C(=O)NCCCCC(C)NC(C2CCOC2C)=O)CC2(C1)CC2(F)F C1(C(=O)OC)CCN(C(c2cc(CNC(=O)CSCCC(C)C)ccn2)=O)C1C N1(C(C(=O)N(CC)CC)=O)CCCC(NC(c2ccc(OC)cn2)=O)C1 N1(C(C2CC(NC(c3scc(C(C)C)n3)=O)C2)=O)CCn2ccnc2C1 C(=O)(C1CSc2ccccc21)NCC1(NC(Cc2nc(OC)sc2)=O)CCC1 c1(NC(=O)COCCC(N2CCC(C(C)(C)C)C2)=O)ccccc1CC1CC1 c1(OC)c(C(N2CCC(C)(C)CC2)C(=O)NCCN2CCOCC2)cc(C)cc1C CC1C(NC(=O)CCC2OCCO2)CCCN1C(=O)Cc1cncc(Br)c1 Cc1cc(C)c(C(N2CCCC2CN(C(=O)C2=NOC(C)C2)C)=O)c(C)c1 c1(C(=O)O)c[nH]c(=NC2CCC(CNC(C3CC3c3ccc(F)cc3)=O)CC2)cn1 c1(OC(C)C(=O)NCCCN(C(=O)Cc2cncs2)c2cccs2)ccc2c(c1)CCC2 N1(C(Cc2cnn(C)n2)=O)CCC2(CCC2NC(c2ccc3c(c2)CC3)=O)CC1 c1(C(N2CCCC3(NC(CC=C(C)C)=O)C2C3)=O)ccc2cncn2c1 C1(C)(C(=O)NC2(CNC(C(c3cn(CC)nc3)=O)=O)CC2)CCC(=O)N1 Cc1ncc(N)cc1C(=O)NCC(O)CNC(c1oc(Br)nc1C)=O Cc1cc(OCC(=O)N(C2CN(C(=O)CSc3cccs3)CC2O)C)cc(C)c1 Cc1cc(N(C)CCC(C)(C)C)nc(=NCC23CCCC2OCC3)[nH]1 c1(C(c2n(CC=C)nnn2)NCC(C)SC)ccc(-c2cccs2)cc1 Cc1ncnc(C(N2CC(NC(=O)C=CC3CCCC3)CC(O)C2)=O)c1C c1(C(N(CCCNC(=O)C(C)C(C)(C)C)CC)=O)cc(C)c(C)c(S(N)(=O)=O)c1 c1(CC)cccc(C(N2CC(CNC(=O)CC3(C)CC3)C(O)C2)=O)c1 C12(C(=O)NCc3cc(C(=O)NC4(CCCC)CC4)n[nH]3)CC(C#N)(C1)C2 N1(C(Cc2c(C)nc(C)s2)=O)CC(CO)C2(C1)CN(C(c1nnc(C)s1)=O)C2 C(=O)(C(CNC(=O)C(C#N)C(C)C)C(C)(C)C)NC(COC)CCO C12(C(N3CCC(C(=O)OC)C3C)=O)CCCC1CCN2C(C1COCCO1)=O c1(C(=O)OC)cc(C(=O)N(CC(C)CNC(=O)C(C)(F)CF)C)c(C)s1 C1(C(C)(F)F)CCN(C(=O)C(=O)NC2CCC2(C)C(=O)O)CC1 c1(C(=O)NC(C(C(C)C)C)CNC(=O)C(=O)N(C)C)ccc2n[nH]cc2c1F N1(C(=O)COCc2nc[nH]n2)CCCC2(C1)CN(C(=O)CC1CCCC(O)C1)C2 N1(C(c2ccc(C(C)(F)F)cc2)C(=O)NCC=C)CCC(O)(CC(N)=O)CC1 C1(C(=O)NCC2C(C(=O)NC(CC)CN(C)C)CC2)C2CN(C)CC12 N1(C(CC2(NC(C3CC(CCC)C3)=O)CCC2)=O)CCCC(C(F)F)C1 c1(CCCC)ccc(C(N2CC(OC)C(CNC(=O)CC3CC(C)C3)C2)=O)cc1 C=CC(C)NC(=O)NCCC1CC1C(C)(C)C C(=O)(CCN=[N+]=[N-])NC(C1CCN(C(C(=CC2CCCC2)C)=O)C1)C CC1CCCN1CCNC(=O)CC1(C)CN(C(C2CC(OC3CC3)C2)=O)C1 C1(CNC2CC3(C(OC)CC3)C2)CCC(C)N(C(=O)OC(C)(C)C)C1 C(CCN(C)C(c1cnnc(C)c1)=O)(C(C)(C)C)NC(C(COC)COC)=O CC1CC2CN(C(=O)CC3CCCN3C(C3CC4CCCC4C3)=O)CC12 C12(C(=O)NCCC(C)CCNC(=O)C3=CCCC3)CCC(CC1)CO2 Cc1c(NC(=O)NC2CC(CNC(=O)CC(C)c3ccccc3)C2)cccc1Cl c1(C(N2CCC(N(C(=O)Cc3cn(C)nn3)CC)C2)=O)ccc(N)c(Cl)n1 C=C(C)CC(C(=O)Nc1cnn(CC)c1)NC(=O)Cn1cc(CC)nn1 c1(CC)cc(C(=O)NCC2(CNC(=O)C(C)CC)CC23CCC3)sc1C C12(NC(Cc3c(C)non3)=O)CCOCC1CN(C(C1C(C3CC3)C1(F)F)=O)C2 N1(C(C2N(C)CCOC2)=O)C2CCC1CC(NC(c1coc(C#N)c1)=O)C2 c1(C(=O)NCC2(C)CCN(C(CSC(C)(C)C)=O)CC2)cc2ccc(Cl)nc2s1 c1(OC(CNC(COC)=O)CNCc2cn(C(C)C)nn2)ccccc1F CCCCCC(CC)C(=O)N1CC(NC(=O)CCCCCCSC)C(O)C1 N1(C(CCOC(C)C)=O)CCOCC(NC(C2COCOC2)=O)C1 N1(C(C(C(=O)OCC)F)=O)CCC2(CC2NC(=O)CCc2cnc[nH]2)C1 C1(=CC(CC)C)CN(S(=O)(=O)CC2CC(C(=O)O)C2)C1 c1(C(N(CCC)CCNC(=O)C(C)(F)C(C)(C)F)=O)ccc2c(c1)CNC2=O Cc1c(F)ccc(C(=O)NCC2CN(C(=O)Cn3cnnn3)C(C)(C)C2)c1Cl Clc1nccc(C(c2nnnn2C2COC2)NC2CC3(C2)CC32CC2)c1Cl N1(C(CSc2c(C)cccc2)=O)CC2CC(C1)CN(C(C1C(C)(C)C1(F)F)=O)C2 Cc1c(NCC(=O)Nc2ccc(F)c(F)c2)ncnc1NC1CCC(C)N1C N1(C(C2CCN(C(CNC(CCC)=O)=O)C(CC)C2)=O)CC2(C1)CN(C)CCO2 CS(=O)(=O)c1cccnc1C(=O)NC1CCC1NC(=O)CCCS(N)(=O)=O S(=O)(=O)(c1cnc2ccc(F)cc2c1)NC1CCC(C(=O)OC(C)(C)C)CC1O c1(SCCC(=O)NCC(C)NC(=O)CCc2nc(=N)[nH][nH]2)ccc(F)cc1 C1(C(C)(C)NC(C2CC(F)C2)=O)CCN(C(c2cc(CO)ccn2)=O)CC1 C1(CCOC)(NC(c2ccn(C(C)C)n2)=O)CCN(C(=O)C(C2CCC2)OC)C1 N1(C(c2c(C)cc(C)s2)=O)CCC2C(C(=O)NCCCC(=O)N(C)C)C2C1 C(CCF)(C(=O)NC1CCCOC1)NC(CCCOCC=C)=O C1(C(N(C)Cc2cc[nH]n2)=O)CCCCN(C(c2n[nH]cc2Cl)=O)C1 CCCC(CC)CC(=O)N(C1CCN(C(=O)Cn2ccnc2)C1)C C=CC(C)(CC)C(=O)NC1CN(C(=O)Cc2cc(Br)cs2)CC1SC C(=O)(C1=NOC(C)C1)N1C2C(NC(c3c(C)n(CCN(C)C)nc3)=O)C(C2)C1 N1(C(C(C)NCC2CCC(C)C2)C=O)CC2(C1)CN(C(=O)OC(C)(C)C)CCO2 C(=O)(C(F)CCC(C)(C)C)NCC1(F)CCN(C(C2C(C(=O)OC)CC2)=O)CC1 C(=O)(C1=CCN(C(=O)C(O)C2CC2)C1)N(CC(C)OC)CC c1(CN(CCNC(c2c(C)nco2)=O)C2CC2)cccc(C)c1OC(F)F c1(C(N2CCCC(CN(C)C(C3CCCS3)=O)C2)=O)cc2n(n1)CCOC2 C12(C(=O)NCC3(CNC(C(C)=C(C)C)=O)CC34CCC4)CCC(C(F)F)(CO1)C2 C1(C(N2C(CC(N)=O)COCC2)=O)CC(F)(F)CN1C(c1scnc1Cl)=O N1(C(COCCOCCOC)=O)CCC(CO)C1C.C1(=O)CCN(C)CCN1 c1(C(c2nnnn2CC(F)F)(C)NC2CCC3(CC3)C2)ccc2c(c1)CCO2 S(=O)(=O)(c1ccc(N2CC3CCC(CO)CC3C2)c(Br)c1)N(CC)CC c1(C(N2C(CNC(C=C(CC)C)=O)CC2)=O)sc(-c2cnn(C)c2)nc1C N1(C(C2CCSCC2)=O)CCn2cnc(-c3ccc(O)c([N+](=O)[O-])c3)c2C1 C1(C(=O)NCC2(CCOC)CCC2)(NC(c2cncn2C)=O)CCCC1C N1(C(COC2N(C(C(C)OCCOC)=O)CC2)=O)CC2(COC(=O)N2C)C1 CCC(C#N)(CC)C(=O)N1CCC(C)(CNC(c2ccccc2Br)=O)C1 C(c1cccc(CO)c1)=CC(N1C(CNC(c2cc(C)sn2)=O)CCC1)=O C(CC1CCCCN1)(C(F)(F)F)NCC1CN(C(C2CCCO2)=O)C1 Cn1cc(C(c2nnnn2CC2CCCO2)NCc2n[nH]cc2C2CCC2)cn1 C1(C(=O)Nc2cn(CCOC)nc2)CCCCN1C(=O)Cc1cccnc1Cl Cc1nn2c(C(=O)NC3CN(C(C4(C#N)CCC4)=O)CC4(CC4)C3)c(C)nc2s1 C1(C(N(CC(CN(C)C(c2sccc2C(N)=O)=O)O)C)=O)(CO)CC1(F)F c1(OC)ccc(Cl)cc1CC(=O)NCC1CC1NC(c1n[nH]c(C)n1)=O N#Cc1cccc(CN(C2CC2c2ccc(OC(F)F)cc2)CCO)c1 C1(NC(C2N(C(C(C)Cn3cccn3)=O)CCCC2)=O)CC2CCC(C1)C2O CN1CCOC(C(=O)NC2CN(C(=O)C(C)(C)CF)CC2O)C1=O c1(C(N2C(C(=O)NCc3ccccc3F)CC(=C)C2)=O)cc(F)c(F)c(Cl)c1F C1(NC(CS(C)(=O)=O)=O)CN(C(=O)CC2OCCC2(C)C)C2CCCC12 c1(C(C(=O)N2CC(CCNC(Cc3cc(C)ns3)=O)C2)(C)C)ccc(F)cc1 Cc1cnc(C(N2CC(O)(C(C)NC(c3ccccc3C(C)O)=O)C2)=O)nc1 C1(O)(CNC(CCCOC)=O)CC2CCC(C1)N2C(=O)CC(C)c1cnn(C)c1 c1(NC(c2cc(C)n(C3CCC3)n2)=O)cc(C(F)(F)F)ccc1Br C1(CNC(c2c(-n3c(C)ncc3)nccc2)=O)CCCN(C(=O)C(C)O)CC1 C(=O)(C1=CC(O)C(NC(=O)CCc2nc(O)n[nH]2)C1)N1CC(C)CC(CC)C1 C1(CC(=O)NC(CC(=O)OC)C2CC2)CC(F)CN1C(c1nc(Cl)cs1)=O c1(C(=O)NCC(CCOC)NC(C2C(C=C)C2)=O)[nH]c2ccc(F)cc2c1Cl C1(O)(CC(=O)NC2(C)CC(NC(CC3OCC(C)(C)C3)=O)C2)CCCCCC1 N1(C(C=C(C)C(C)C)=O)CCOCC(NC(=O)C(C)CC(N)=O)C1 c1(C(N2CC(NC(C3CCCCN(C(=O)C4CC4)C3)=O)C2)=O)cccc2nncn12 Cc1sc(C(N2CC(CNC(=O)CC34CCCC3C4)CC(C)C2)=O)c(C)c1C CC(CC(=O)NCC(C)(C)CC1CN(C(C2CCCC(C)C2)=O)C1)CC(C)(C)C C1(NC(C(N(C)C)C2CC2)=O)CN(C(C2CC(=O)C2(C)C)=O)CCC1O C1(C(=O)N(c2ccsc2)Cc2ccc(Cl)c(Cl)c2)COc2ccccc2O1 c1(CCNC(CC(C2CC2)NC(C2C(CC)CCC2)=O)=O)cn(C)nc1C c1(C(C)F)ccc(C(N2CC3CC2C3NC(=O)CN2C(C)CCC2C)=O)cc1 C1(NC(C(C(F)(F)F)OC)=O)(CNC(=O)C(C)(C)OC)CC2CCC1CC2 C1(NC(Cn2ncn(C)c2=O)=O)CN(C(C2CCCCCC2)=O)CC1N=[N+]=[N-] C(=O)(C(C)C(=O)NCC(N1CC(C)CC1CO)=O)OC C#CCCC(=O)NC1CCCC1NC(c1cc[nH]c1C1CCCC1)=O C(=O)(C(C)(C)CC(C)C)N1C(C)CCC(NC(C=C(C)I)=O)C1 C1(NC(=O)CC2CC2(Cl)Cl)CCC(NC(c2cnco2)=O)C1 C(=O)(C1=C(C)OCCS1)N1CC(CC)C(NC(c2ccc(F)cc2C#N)=O)CC1 Cc1nc2n(n1)CCN(C(=O)C(C1CCN(C(C3C=CCS3)=O)CC1)C)C2 C1(NC(C(C)(C)F)=O)CC2(NC(=O)Cc3c(Cl)cccc3Cl)COC1C2 CC1OC2(CNc3cc(Cl)ncn3)CC1(NC(=O)C(=O)NCCC(N)=O)C2 N1(CC#CC)CCC2C(NC(=O)CCc3ccsc3)C(C)(C)C12 N1(C(=O)OCC)CCC(CC(C)SC2C(NC(c3c[nH]nc3C(C)C)=O)C2)CC1 Cc1csc(C(=O)NCc2ccc(C(C)NC(=O)C(C)NC=O)cc2)c1Cl c1(N2CCC(C(F)F)(CNC(=O)C3=C(Cl)CCOC3)C2)ccc(F)cc1[N+](=O)[O-] CN1CC(C(=O)NC2CC(NC(=O)C(C3CC3)C3CC3)C2)C(C(F)(F)F)C1 Clc1cccc(CNC(=NCC2CCCC2)NCC23CC(CO2)C3)c1 C1(NC(CCCOCCC)=O)CN(C(=O)C(C)CC(C)C)CCC12CCOCC2 c1(C(C)NC(C(CC=CC)NC(=O)Cc2ccn(C)n2)=O)ccc(F)c(F)c1 c1(CC(=O)N(C(CCNC(CC=C)=O)C)C)cn2cc(C)sc2n1 C#CC1(O)CC(C(=O)NCC(C)(C2CC2)NC(=O)CC(O)C2CCCC2)C1 O=Cc1cccnc1-c1ccc(C(=O)NC(c2ccsc2)CO)s1 C(=O)(C1=CSCCO1)N(C(C)CCNC(c1ccc(OCCF)cc1)=O)C C(=O)(C(F)C(F)(F)F)N(C)Cc1c(CNC(C(COC)(C)OC)=O)cccc1 c1(OC)n[nH]cc1C(=O)NCCCCCNC(C1CC(c2ccccc2)CO1)=O C1(OC)CC(CNC(c2cc[n+]([O-])cc2)=O)N(C(=O)C(C)Oc2cccnc2)C1 O=C1NC(=O)C(C2CN(c3ccc(-c4cc[nH]n4)s3)C2)N1 C1(CNC(c2c(C)ccnc2)=O)CCC(C)N(C(=O)CC2CCOC2)C1 N1(C(C(C)CF)=O)CCOC2(CCCN(C(c3cc4n(n3)CC3(CC3)C4)=O)C2)C1 c1(C(N2CC3CCCN(C(CCC#C)=O)C3C2)=O)cccc2c1OCC(=O)N2 c1(OC)ccc2c(CC(=O)NCCNC(C3(C)CCC(C)C3(C)C)=O)c[nH]c2c1 c1(C(N(C(C)C(=O)Nc2cn(C)nc2O)C)=O)cccc(O)c1F C1(C2(O)CCC(=O)CC2)(C(=O)NCCc2nc(N(C)C)sc2)CC1 c1(C(N2CCC(NC(C(CC(=C)C)OC)=O)CC2)C)ccc2c(c1)OCO2 N1(C(C(COC(C)=O)C)=O)CC=CC(NC(=O)CSc2cnn(C)c2)C1 C1(OC)CC(CNC(=O)COc2cccc(F)n2)N(C(c2cnc(C)n2C)=O)C1 C(=O)(N1CC(O)CCO1)C1CCN(C(C2CC2F)=O)CC1 C(N=c1ccnc(Cl)[nH]1)C1C(C)CCN(C(c2c(C)noc2C)=O)C1 CN=C(NCC1CC1c1ccc(C(F)(F)F)cc1)N1CCC(c2ccccn2)C1 C12(C(=O)NC3CC(NC(C4C(C(N)=O)C4)=O)C3)CC3CC(C(=O)N1)C2C3 C1(C(N2CC(CNC(C(COC)N(C)C)=O)C2)=O)CC2OC1C1CC21 N1(C(c2[nH]cc(CC)c2)=O)CC(CO)C2(C1)CN(C(=O)Cc1cc[nH]c(=N)c1)C2 c1(CC)nn(C)cc1C(N1CCOCC1CC(=O)NCCCc1cn[nH]c1)=O Cc1ccc(C)c(C(=O)NCC2OCCC2C(N2CCCCC2C(C)(C)O)=O)n1 c1(OC)cccc(N2CCC(F)(c3ccccc3)CC2)c1[N+](=O)[O-] c1(CNC(CCn2cc(CC(C)O)nn2)=O)ncccc1Oc1cccc(F)c1 c1(C(N2CCCC(C)(O)C2)=O)ccc2c(c1)CN(C(=O)C=Cc1cnc[nH]1)CC2 C1(O)(CN(C(c2cc(OCC)n[nH]2)=O)C)CCCN(C(=O)C=CCF)C1 Cc1c(C(=O)NCCCOCCN(C)C(C2CCS(=O)(=O)N2)=O)cnn1C N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C(C2C3CCC(=O)C23)=O)CC12CC2 C(=O)(C1CCSc2ccccc21)N1CC(OC)C(NC(=O)CCn2cncn2)C1 C12(CN(C)C(C3CC(n4cc(-c5cn[nH]c5)nn4)C3)=O)CC3CC1C2C3 C1(C(=O)NC(c2nccc(O)n2)C)CCC(C2CC2)N1C(C1CC2(CCC2)C1)=O c1(C(=O)NC2C(CNC(CC(C)OC)=O)CC2)sc(N2CCCC2)nc1C c1(N(CC(C)C)CCS(=O)(=O)CC2CC(O)CN2C)ccccc1Cl C12(CNC(C(C)Sc3ccccc3)=O)CC(C1)C(NC(=O)CNC(N)=O)CO2 C1(CNC(CN(S(C)(=O)=O)C)=O)(NC(=O)CC2CC23CC3)CC2CCC1CC2 CCCC(C(=O)NC1CCN(C(C2(OCC)CCC2)=O)C1)N(C)C C(=O)(C(CNC(=O)Cn1cc(Cl)cn1)CC(C)C)N1CCC(C)(CC)C1 N1(C(CC(CNC(C(C)NC(C)=O)=O)C)=O)CCC2=C(CCCC2)C1 N1(C(C=C(C)C(C)C)=O)CCN(C(c2ccccc2)=O)CC(C)(F)C1 S(=O)(=O)(c1ccc2c(c1)CCCC2)NCCc1cc(OC)cc(OC)c1 c1(C(C)C)ccc2cc(C(=O)NC3CCC(CNC(=O)COC(F)F)C3)[nH]c2c1 c1(CC)ccc(C(=O)N(C)CCN(C(=O)Cc2ccno2)C)cc1CC C1(NC(c2cccnc2)=O)CCC2(CCNC2)CC1 C=CC(C)(O)C(=O)N1CCC(c2cc(CNC(C3CC3(C)C)=O)on2)CC1 CN1N=CC(CC(=O)NC(CNC(c2cc(C3(Cl)CC3)n(C)n2)=O)CO)C1=O C1CCCC(CNCC(N2CCCC2)C2CCCO2)CCOC(OCC2CC2)C1 c1(CC(=O)N(C(CN(C(C(c2nc(C)sc2)=O)=O)C)C)C)cc(C)nn1C c1(C(N2CC(N(C(C(C)SC)=O)C)C(O)C2)=O)ccc2c(c1)OCCO2 CCCN=C(NCC1CCCC(OCC)C1)N1CCC2(CCOC2)C1 C1(C(=O)NC(C)(C)CC(F)F)CCN(C(=O)CCC2CCCCO2)C1(C)C c1(-c2cncc(CO)c2)ncn2c1CN(c1ccn3ncc(I)c3n1)CC2 c1(NC)ccc(C(=O)NC(CC(=O)NC2CCOC2)C(C)C)cc1C c1(OCC)cc(C#N)ccc1CN1CCOC(CC(=O)NC2CCC(=O)NC2)C1 O=C(CCCCCCBr)NCC1CCC(C(=O)NCCc2ccc(F)cc2)CC1 C1(C(N2CC3(C(NC(C4CC5(CCC5)CO4)=O)CC3)C2)=O)Cc2ccncc2N1 c1(C(=O)NC(C)C#N)cc(N2CCOCC2)ncc1Cl c1(C(N2C(C)CC(NC(C3CCC(N(C)C)CC3)=O)C2)=O)ccn2ncnc2c1 c1(COC)cccc(C(=O)NC(C)C(C)NC(C2CCCC2O)=O)c1 c1(C(N(CC(C)NC(=O)CC2CC(=O)NC2=O)CC)=O)ccc2c(c1)CCOC2 CCC(C)C(C)C(=O)NC1CN(C(c2ccc(CNC(N)=O)cc2)=O)CC1(C)C CC(C)CC(CNC(c1nnn(C)c1N)=O)NC(=O)CSCc1cscn1 Cc1cc(C(N2CCCC(C)(C(=O)NCC3([Si](C)(C)C)CC3)C2)=O)nc(C)c1 N1(C(C2N(CC)CC2)=O)CCC2(CCCN2C(c2[nH]cc3c2CCCC3)=O)C1 CCCCC(C)C(=O)N1CCCC(N(C(c2ncccn2)=O)CC)C1 c1(C(=O)NC(CCCNC(c2cn(CCC)nn2)=O)C)cc(C(N)=O)ccc1C n1(CC)ncc(Br)c1C(N1CC(N(C)C(C2CCCS2(=O)=O)=O)C1)=O CC1(C)CCC(NC(=O)Cc2ccns2)C(CNC(c2ccc(Cl)nc2N)=O)C1 C1(NC(C2C(OC)CC2)=O)CC2CCC1N2C(c1cscc1Br)=O c1(CC)ccc(C(=O)NCC2CC2NC(C2CCCO2)=O)cc1Br C(=O)(CCC(C)(F)F)NC1C(C2CCN(C(C=CCOC)=O)CC2)OCCC1 O=C(C(CC(F)(F)F)c1ccc(F)cc1)NC1CCC1NC(=O)C1=CCCOC1 CC(CN(C)C)CCC(=O)N(CC(C)(C)CNC(C1(CN(C)C)CC1)=O)C C1(NC(COCCCC)=O)CCC2CC1CN2C(c1cncc(C2CC2)n1)=O N1(C(C(C)C)=O)C2CCC1C(CNC(c1ccc(OCC3CC3)cc1)=O)C2 N1(C(c2c(C)nnn2C)=O)CC2(CC(NC(=O)C(CO)C(C)C)CO2)C1 CC#CCCCC(=O)N(CCN(C(=O)CNS(C)(=O)=O)C)C(C)C CCC(C)(O)C(=O)N1CCC(C(C)(C)NC(C2CN(S(=O)(=O)CC)C2)=O)CC1 C1(C(=O)NCCCC(C)NC(C(C)N(CC)CC)=O)COCCN1C=O N1(C(C(CC)Cc2cccc(C)c2)=O)CC2CC(C1)C2NC(=O)C(C)CCOC C(=O)(CC(C)C(C)(C)NC(=O)CSCCCC)N(CCC#C)C c1(-n2ccc(C)n2)cccc(NC(=O)C(C)Oc2ccccc2F)c1 CN1N=C(CC(=O)NC(CNC(C2CNC(=O)N2)=O)C2CC2)CC1=O c1(C(N(C2CN(C(=O)C(C)(C)CF)CC2O)C)=O)ccc(C2CC2)cc1F CCCC(O)(CCC)CC(=O)N1CC(F)(CNC(C2CC2(C)Br)=O)C1 N1(C(=O)OC)CC(NC(=O)CNC=O)C1.C12CCC1C(=O)N2 Cc1sc2ncc(C(=O)NC3(CCNC(C45CC6CC4C5C6)=O)CCC3)n2c1C N1(C(c2ccnc(F)c2F)C(=O)NC)CCC2(CCN(C(C)=O)C2)C1 C1(C(=O)NC2CC(NC(C(C)OCc3ccc(F)cc3)=O)C2)CC2C=CC1O2 CC1CC(C(=O)OC(C)(C)C)CN(C(=O)C(C)(C)NC(C2CC23CC3(F)F)=O)C1 c1(C(=O)NCCC(C)NC(CCC2C(C)=NNC2=O)=O)ccc2ncsc2c1 C=C(C)C(C)(C)C(=O)NCC(C)(C)CCNC(C1CCN(C2CC2)CC1)=O CC(C(=O)NCCn1cc(CNC(C2(CF)CC2)=O)nn1)C(C)S(C)(=O)=O CN1CCN(C(C2COCC2(C)C)=O)CC1C(N1CC(O)C(O)C1)=O C1(CNC(CC(C)(C)C)=O)CC2(CCN(C(=O)CC3CCCO3)CC2)CO1 N1(C(CC(C=C)(C)C)=O)CCC2(CCN(C(c3ccnn3CCCC)=O)C2)C1 Cc1cc2scc(CC(=O)Nc3ccccc3OC(C)(C)C)c2s1 C1(CCC)(NC(=O)C=CC=C(Cl)Cl)CCCN(C(=O)C(c2ccc(C)cc2)C)C1 N1(C(c2c(C)csc2)=O)CC(CNC(c2[nH]cnc2C)=O)OC(C)(C)C1 c1(CC(=O)NCCNC(C2CN(C)C(=O)C2)=O)c[nH]c2ccc([N+](=O)[O-])cc12 C1(CC(=O)NCC2(C(=O)NCC(COC)(C)O)CC(F)C2)CCC(=O)C1C c1(C(N(CCCNC(C(CC=CC)C)=O)C)=O)[nH]c(C)c([N+](=O)[O-])c1C N1(C(CCC=C)=O)CC(NC(=O)Cc2ccccc2C)C(C2CC2)C1 c1(C(C(=O)O)NC(c2n(C)ncc2)=O)cc2ccccc2o1.C1CC1 N1(C(C(CCSC)NC(C)=O)=O)CCC2(NC(C3C=CCCC3)=O)CCCC12 c1(C(=O)NCC2N(C(C(C=C)(C)CC)=O)C3CCC2C3)nc(O)nc(O)c1F C1(CNC(C2CC2(Cl)Cl)=O)CCN(C(C23CCCCC2C3)=O)CC1 c1(C(N2CCC(c3ccnn3C)C2)C(=O)OC)cc(C(F)(F)F)cc(F)c1 C(=O)(C#CC1CCCCC1)NC(CC)CNC(c1cc(C#N)ccc1Br)=O c1(CC(=O)NCC2C3CN(C(C4CC4(F)F)=O)CC23)c[nH]c2ccc(Br)cc12 c1(C(=O)NC2CN(C(C(C)OC)=O)CC2(C)C)coc2ccc(C)cc12 c1(OC)ccc2ncc(C(=O)NCCCCN(C(=O)CCNC(N)=O)C)n2n1 c1(CN)ncn2c1NC(=O)C(CC(=O)NC(C1CCOC1)C1CCC1)C2 C1(CC(=O)NC23CCC(C2)N(C(c2cnns2)=O)C3)SC2=NCCN2C1=O c1(CC)c(C(=O)NCC2CCC2CNC(c2cc(O)nc(Cl)c2)=O)cccc1F c1(N2CCC(C)(COC)CC2)[nH]c(=NCC2CCC=CO2)nc2scnc12 c1(CC)cnccc1C(=O)N(C)CC1(O)CCN(C(C2CC2F)=O)C1 C(=O)(C(CC(C)C)NC(=O)OC)N1CC(C(=O)Nc2c(CC)nns2)OCC1 c1(OC)ccccc1C(CNC(C1CCCCS1)=O)NC(=O)Cc1ccsc1 CCC(C)CCC(=O)N1CC(CNC(c2ccc(C)c(OC)c2)=O)C(O)C1 Cc1nccc(C(N2CCC(C(C)NC(C34CC(C3)S(=O)(=O)C4)=O)CC2)=O)c1N C1(C(N2CC(C(=O)N(C)Cc3ccnn3C)(SC)C2)=O)CC2(CCC2)C1 NC(C(=O)N(CCO)C1CC1)c1cscn1 N1(c2cc(N(C)Cc3ccc(CC)o3)ncn2)CCC2(CC(=O)N(C)OC2)C1 c1(CC(c2nocc2C)NC(=O)NC(CC#C)C)cccc(Br)c1 N1(CC(N2C3CN(C(C(C(CC)O)C)=O)C(CC3)C2)=O)Cc2ccccc2C1=O CC1CN(C)CC(C(=O)NC(C(=O)NC2CC(=O)NC(=O)C2)C2CC2)O1 c1(C(=O)NCCCNC(C(=O)NC(C)C)=O)ccc2c(c1)CN(C)CC2 C1(CC(=O)NC(c2ncc(C)o2)C)CCCN(C(c2coc(C)n2)=O)C1 C12(NC(=O)NCCC3CCC4CC34)CCCN(CCC1)C2 Cc1cc(C(=O)N(CCN(C(=O)C=CCO)C)Cc2ccccc2)no1 Cc1ccc(F)c(C(=O)NC(C)CCCCNC(=O)CC23CCC(CC2)C3)c1F CC1CN(C(c2cnsn2)=O)CCC1CNC(c1cccnc1)=O.C1(=O)CN1 C(=O)(CCC1=CCc2ccccc21)NC(C1OCCN(C(CC)=O)C1)C Cc1ccc(C#N)c(N2CCC(O)(C(C)NC(=O)C(C)C3CCOC3)CC2)n1 C1(C(C(C)NCCN(C2CC2)CCCN)OC)CCCC(F)(F)CC1 N1(CC(=O)NCCC(=C)CNC(=O)CC(C)CC(C)C)CCSC2CCCCC12 c1(CC)noc2ncc(C(=O)NCCC(C)NC(c3c(C)ccnc3O)=O)cc12 N1(C(CC=C)=O)CCC2(CC1)OCCCC2NC(=O)CC1=NNC(=O)C1 C(=O)(CC1=CCN(C(=O)Cc2ccc(F)nc2)CC1)N1CC(CC(=O)OCC)C1 c1(C(=O)NCC23CC(NC(C(C(C)C)n4cnnn4)=O)(C2)C3)cc(N)ccc1Cl CC1CC(C)N(C(=O)CCc2nc[nH]n2)CCN1C(C1CCC(C(F)F)CC1)=O C1(NC(=O)C2=CCCC2)CS(=O)(=O)CC1NC(C1CC(C(F)F)C1)=O N1(C(C=CC(=O)OCC)=O)CC2COCCC2(NC(c2n[nH]c3c2COC3)=O)C1 c1(CCC(=O)NCC(CC)NC(=O)CSCC#N)ccc(OC(F)(F)F)cc1 CC1CN(C(=O)C(c2ccc(Cl)s2)=O)CC(c2ccccc2)O1 Cc1cccc2nc(C(=O)NC3CCCCNC3)cn12 CC(C)CC(C)C(C)NC(C1CN(c2ccc(C#N)nc2)C1)=O c1(N2C(C3(C)CC3)CSCC2)nc(=NCC(C)(C)F)[nH]c2c1COCC2 c1(CNC(C(=O)NC(C(CC)CC(C)C)C)=O)ccc2nnc(S)n2c1 c1(NC(C(C(=O)OC)C)=O)cc(C(=O)NC2(CN)CC2)ccc1Cl Cc1cc(O)n2ncc(C(N3CC4CCC3CN4C(C3CSC3)=O)=O)c2n1 Cc1cnccc1C(=O)NC1CC(CNC(=O)CC(C)(C)C2CCCCC2)C1 c1(CCCC(=O)N(CC(C)CNC(c2cnc(C3CC3)[nH]2)=O)C)ccccc1N C(CCCCC(=O)NC1CC=C(C(=O)NC2CCC(F)(F)C2)C1)SC C1(C(C)(C)OC)CCCN(C(c2cn(C)c(-c3ccccn3)n2)=O)C1 c1(CNC(CCn2cc(-c3ccc(C(N)=O)cc3)nn2)=O)ncc(F)cc1F C1(O)(CNC(C(COCC)C)=O)CCCN(C(=O)C(C)Cc2cccc(F)c2)C1 c1(CC(N2CCC(NC(C(C)CO)=O)C2C2CC2)=O)ccc2c(c1)CC2 C1(C(=O)OC)=C(C(F)(F)F)C(NC(=O)NCc2cc(C(=O)OC)n[nH]2)CCN1C Cc1nnc2n1CC(C(=O)NC(C)CNC(c1cnn(CCOC(C)(C)C)c1)=O)CC2 C12(C(=O)NC(C3CCCN3C(=O)CN3CCCCC3=O)C)CC(C1)C(C)O2 CC1CCOC(C(=O)N(C)CC2CCN(C(=O)CC3CNC(=O)O3)CC2)C1 c1(C(N2CCCC(C)(C)C2)C(=O)NCCOCC2CC2)cccn2ccnc12 C(=O)(CC(C)(C)CC(=O)N(C1CCCCN(C(c2n[nH]c(C)c2F)=O)C1)C)OC n1(CC(N2CC3C(CNC(C(CC)C)=O)(C3)C2)=O)ccc([N+](=O)[O-])n1 c1(C(N2CC(OCCNC(c3ncc(C#N)nc3)=O)C2)=O)cc2ccnc(Cl)c2[nH]1 Cc1cnccc1C(N1CC(NC(=O)C(C2CCOCC2)C)C(C)C1)=O C1(NC(c2c(C)cc(C)[nH]2)=O)CC2CN(C(c3ccc(F)c(C)c3)=O)CC2C1 C1(C(=O)NC2CC(C#C)C2)(OC)CCN(C(C2CCC(N(C)C)C2)=O)C1 c1(NC(C23C(NC(CSC)=O)CCC2C3)=O)cc(F)c(F)cc1C C1(OC(C)C)CC(N=c2[nH]c(=NCC3(C)CCN(C)C3)[nH]c3c2CCCC3)C1 CC1(C)C=C(C(=O)NCC2(C)CCN(C(=O)C(N3CCOCC3)C3CC3)C2)C1 c1(OC)cnnc(C(=O)NC2CCC(C(=O)N(CC(=O)N(C)C)C)CC2)c1 c1(C(=O)NCCC2(O)CN(C(c3cn4c(n3)SCC4)=O)C2)ccc(O)c(CO)c1 C1(NC(C2C(C(=O)OC)C2)=O)CC2CCC(C1)N2C(c1cc(F)c[nH]1)=O C1(O)(CN(C(C(n2cc(Cl)cn2)C)=O)Cc2ccccc2)CN(C(=O)CC2CC2)C1 C(CCC(C)(C)C)(C(N)=O)NC(C(=O)Nc1cnc(C(C)C)[nH]1)=O Cn1cnc2c(C(N3CC(NC(=O)CCCC#N)CCC(O)C3)=O)[nH]nc2c1=O Cn1ncc(C(=O)NC(CNC(=O)CCC2NC(=O)NC2=O)CO)c1S(C)(=O)=O c1(CCC(N2CCCC(C(N(CCCC)CCO)=O)C2)=O)cc(F)cc(F)c1 c1(C(=O)NC2C(CNC(c3c(C)cnn3C)=O)CC2)ccc(F)c(F)c1 C1(CNC(C(C(C)C)OCC)=O)CCN(C(C23CCCC2CCC3)=O)CC1O C1(=CCNC(C(CC)c2ccccc2)=O)CCN(C(C2CC(C(F)F)C2)=O)CC1 C(C(O)CN=c1[nH]nc(-c2ccccc2)s1)CC(=O)N(CCCCCC)C1CC1 N1(C(CC#N)=O)CCCC(F)(CNC(=O)C2=C(Cl)CCCC2)CC1 C1(CC(N2CC(NC(C=C(C)C(C)C)=O)CC2(C)C)=O)CC2(CCC2)CCO1 C(=O)(C(C#N)C(C)(C)C)N1CCC(N(CCC)C(C2C=CCC2)=O)CC1 CCCC(C)(C)C(=O)NC12COC(C1)C(NC(=O)C(C)(F)CC)C2 N1(C(C(c2ccccn2)C)=O)CC(F)CC1CNC(C1CCC=CO1)=O C(=O)(CCCCCCS(N)(=O)=O)NC1CN(C(C(CCOC)C)=O)C2(C1)CCC2 N1(C(CCOC(C)=O)=O)CCC2CCC(NC(=O)Cc3cc[nH]n3)C1C2 CC1CC(C(N2C3CCC(C3)C2CNC(=O)Cc2nc[nH]n2)=O)CC(C)(C)C1 c1(C(C)(C(=O)O)NC(C(C2CCCCC2)C)=O)ccc(NC(=O)OC(C)(C)C)cc1 C(=O)(C(CCCO)N(C)C)OCCCCN1CCC(OC)CC1 N1(C(C=C(CC)CC)=O)CCCC(O)(CNC(=O)CN(C)CCOC)CC1 Cc1nc(C(c2nnnn2Cc2nnn(C)n2)NCCCc2ccsc2)sc1Br c1(C(=O)NC(C)CN(C(=O)NC(CC)=O)C(C)C)cn(-c2cnn(C)c2)nn1 C1(F)(CNC(c2cnn(C)n2)=O)CCN(C(=O)CCSC(F)(F)F)C1 C(=O)(CC(C)CC(F)(F)F)NCC1C(C)(C)CCN(C(c2n(CC)nnc2)=O)C1 C(=O)(C(C(C)(C)CC)OC)NC1(CF)CCN(C(c2c(CC)cc(Cl)cc2)=O)C1 C(=O)(CN=S(C)(C)=O)N(CCNC(=O)Cc1cnsc1)CC C1(C(N2CC(NC(c3cc4sccc4cn3)=O)C(O)C2)=O)CC2(C1)CC(F)(F)C2 N1(C(c2sc(CCC)c(CC)c2)=O)CCCC12CCN(C(=O)C#CC1CCC1)C2 c1(OC)cnc(Cl)[nH]c1=NCCC1C(C)CCCN1C(=O)C(C)OC N1(Cc2nnc(C)o2)CCCC(C)(NC(=O)Cn2cc(CN)nn2)C1 c1(OC)ccc2[nH]c(C(=O)NC(C)(CNC(=O)COCCSC)CO)cc2c1 Cc1nn(C)c(C)c1C(=O)NC1CCCN(C(=O)CC(=O)OC(C)(C)C)C1CO C1(C(=O)NC(CNC(C2N(C(C)=O)CCCC2)=O)C)CCN(CCO)C(=O)C1 C(C(C)(COC)C(=O)N1C2CCC1C(C(=O)NC(C)CCN1CCCC1)C2)OC C1(CNC(C2CC(n3ccnc3)C2)=O)CC2CC2N1C(C1CC(F)(F)C1)=O Fc1ccc(F)c2c1CCN(c1nc(N3C4CCCC3CC4)c3c(n1)CCC3)C2 C1(CCC)CN(C(c2cc(C(F)F)ccn2)=O)CC1NC(c1ccc(O)nc1)=O C1(NC(C2N(C(C(C3CC3)OCC)=O)CC(C)C2)=O)CC2CCC1(CO)C2 c1(C(N2CCC(C(CNC(CS(C)(=O)=O)=O)F)CC2)=O)ccnc2ccsc12 C=CC(C)(O)CC(=O)N1CCCOC(CNC(c2ccccc2C2CCC2)=O)C1 S(=O)(=O)(c1cccc(=NC2CCN(S(C)(=O)=O)C2)[nH]1)N1CCCC(C=C)C1 C(=O)(C(C)(C)CS(C)(=O)=O)NC1CC2CN(C(C(CC)OCC)=O)C(C1)C2 C12(CC(=O)NC3C(C)CN(C(C4(F)CC=CC4)=O)C3)CC3CC(CC(C3)C1)C2 c1(NC(CN2C(c3onc(C)n3)CCCC2)=O)cc(F)cc([N+](=O)[O-])c1 CC1OC2(C)CC1(C(N1CCC(c3cn(-c4cccc(Cl)c4)nn3)C1)=O)C2 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC(NC(=O)CCC2(C)CC2)C(C(C)C)C1 C1(NC(C(CCSC)O)=O)(CO)CCCN(C(=O)Cn2cc(N)cn2)C1 C1(C(=O)NCCC2CCN(C(CNC(C3CCCC3)=O)=O)C2)CCCC12CC2 C1(C)(C(=O)NCCCC(C)NC(=O)C(c2ccc(F)cn2)(F)F)CC=CCC1 N#Cc1ccc2c(CN3CCC(C(=O)Nc4cccc(O)c4)C(O)C3)c[nH]c2c1 C(=O)(C(CCC1(C)CC1)N1CCCCCC1)NC(c1nnnn1C)C C(C)(C(C(=O)N1CCC1(C)CCOC)NC(=O)Cc1cn[nH]c1)OC Cc1cccc(C2CCCCN2C(=O)NCC2(C3CCC=CCCC3)CC2)c1C N#Cc1ccc2c(c1)CCN2C(=O)C(C1CCC1)NC(=O)C=C1CCOCC1 C1(NC(C2N(CC)CCC2)=O)CN(C(c2cnsc2)=O)CCC12CCC2 n1(CC)cc(CN2CCC2C(=O)Nc2c(Br)cnn2C)c2cccnc12 C1(NC(CC2(C=C)CC2)=O)COC2(C1)CN(C(c1ccc(-c3cc[nH]n3)s1)=O)C2 Cc1ccc(C(N2CC(NC(c3coc(C(F)(F)F)n3)=O)C3(CC3)C2)=O)c(Cl)c1 Cc1cccc2[nH]cc(CC(=O)NC3CCCN(C(=O)Cc4cnsc4)C3C)c12 N1(C(CNS(CC)(=O)=O)=O)CC(C)CN(C(c2cn(C)nc2OC)=O)CC1C C(CC(C(=O)N1CCC(N(C(=O)C(C)SCCCC)CC)CC1)OC=C)CC=C c1(CNC(C2CN(C(c3ccnnc3)=O)C2)=O)ccccc1Cl c1(SC)cc(N2CCCC2CCCO)ncn1.c1(NC(=O)NC)ccccc1 c1(C(N2C(C(C)NC(C3(N(C)C)CC3)=O)CCC2)=O)cc2cccnc2o1 c1(C(N(CC(C)NC(=O)Cn2cnc(C(F)(F)F)n2)C)=O)ccc(CCF)cc1 C1(O)(CC(=O)N(CCC(C)NC(C2CCC2C(F)(F)F)=O)C)COC(C)(C)C1 C1(NC(C(C)OCCOC)=O)CC(OC)CN(C(c2nn(C)c(C)c2N)=O)C1 C=C(C)C(C)(O)C(=O)N1CCC(O)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(C(=O)NC2(CNC(=O)COC3CCC3)CCOC2)cnn2ncccc12 C(=O)(CS(C)(=O)=O)N1CCC(N(C(c2c(CC)nco2)=O)CC)C1 C1(COC)COCCN1C(=O)C(N1CCC(OC(c2cnn(CCO)c2)=O)C1)=O C1(CCNC(c2cc(Cl)c[nH]2)=O)CN(C(c2ocnc2C2CC2)=O)CCCO1 C1(C2CCCN(C(c3nnn(C(C)C)c3C)=O)C2)(NC(C(CC=CC)C)=O)CC1 c1(C(N2CCC(CN(C)C(C34CCC3C4)=O)CC2)=O)ccc2c(c1)nc(O)n2C N1(C(C)=O)CCCC12CCN(C(C1CCCN(C(c3sccc3Cl)=O)C1)=O)C2 N1(C(C(CC)(F)F)=O)CCC(C)C(NC(c2cc(Cl)ccc2Cl)=O)C1 C12C3C=CC(C3)C1N2.c1(CC(N)C(=O)N2CCCC2)ccc(F)cc1 C12CCCN(C1NC(CCc1ccc(C)nc1)=O)C2=O.C1(C(C)C)(CO)CCC1 CC1CCC(C)N1C(c1cccc(-c2nc(C(F)(F)F)nn2C)c1)=O c1(NC(COC(CNC(C(C(=O)OC)C)=O)(C)C)=O)cc(C)cn(C)c1=O Cc1csc2cc(C(=O)N(C3CCC(NC(=O)C(=O)N(C)C)CC3)C)[nH]c12 Cc1cc(C(N2CC(C)C(NC(=O)Cc3[nH]cnc3C)C(C)C2)=O)c(F)cc1F C1(NC(C2(C(=O)OC)CN(C(N)=O)C2)=O)CCN(C(=O)OC(C)(C)C)CC1C C1(C(=O)NCC(C(C)C)NC(=O)CCc2ccc(N)cc2)CCCCC12CCC2 c1(N2CCCC(CCC)CC2)cc(Br)ccc1S(=O)(=O)NC1(CC)CC1 C(=O)(C(C)(C)S(C)(=O)=O)NC1CC(CNC(c2ccc(OC)c(C)c2)=O)CC1O C(=O)(CCCOC(C1(OC)C=CCC1)=O)OCC CC1=C(C(=O)NC2CC3CCC2N(C(c2c(Cl)nn(C)c2Cl)=O)C3)SCCO1 c1(-c2nc(-c3ncc(CN(c4ccc(F)cc4)CC)[nH]3)on2)ccc(F)cc1F C1(O)(CCNC(C(C)=CC2CC2)=O)CCN(C(c2ccc(CC)[nH]2)=O)C1.COCC C1(O)(CNC(C(C)OCC2CC2)=O)CCN(C(c2cn(C)[nH]c2=N)=O)C1 N1(C(c2cc(C)sn2)=O)CC2(CCCC2NC(c2cncn(C)c2=O)=O)C1 c1(OC)cccc(-c2nnc(Cc3ccc(F)cc3)o2)c1.C(=O)C1CC1 CCC(COC)C(=O)NC(C)CCCNC(=O)COc1cc(C)on1 CC(C(=O)N1CCCC1C1CCN(C(=O)CN2CSCC2=O)C1)C(F)F CCCC(C(O)C(=O)N1CC2(C1)CN(C)C2)NC(=O)CC1CCCCC1O c1(NC(C23CC2CN(Cc2ccc(Cl)nc2)C3)=O)ccc(F)c(Br)c1 C#Cc1cncc(C(N2CCCC(CNC(C3CS(=O)(=O)C3)=O)C2)=O)c1 CCCC(F)C(=O)NC1CCN(C(c2csc3nccn23)=O)CC1 CC(C)(C)C(O)C(=O)NC1CCC(CNC(c2ccc(-c3nnco3)cc2)=O)C1 CCC(C)C(C)(c1nnnn1C1CC1)Nc1cncnc1CC c1(C(=O)NC2CN(C(Cc3ccc(C)cc3)=O)C2)c(Cl)ccc(Br)c1F C(C)(CNC(c1ccncn1)=O)(CC(C)C)NC(c1c(C)nc(CC)s1)=O c1(C(C(=O)N(CCN(C(=O)COCC2CCOCC2)C)C)N(C)C)cncn1C c1(C(N(CCNC(C2CCCSC2)=O)CC)=O)cnc2[nH]ccnc1-2 Cc1cnncc1C(N1CC2C(NC(C3(c4ccccc4F)CC3)=O)C2C1)=O n1(CC=C)cc(C(=O)NCC2CCCC2NC(C2(N3CCOC3=O)CC2)=O)nn1 C#Cc1ccc(C(=O)NC2C=CC(CC(=O)NCc3nnc(O)n3C)C2)cn1 C1(CNC(C(C2CCOC2)OC)=O)CCN(C(C23CCC(C)(C2)OC3)=O)CC1C C1(O)(C(C)NC(c2cnc(C(F)F)s2)=O)CCN(C(=O)C(C)(C)C2CCC2)C1 N1(C(N(C2CCC(=O)NC2)C)=O)CC(O)CC(C)(C)C1 N1(C(CC2CCN(C)C2=O)=O)CCC2CCC(C1)N2C(C1Cc2ccccc2C1)=O CC1CN(C(=O)C=CC(=O)NC2CC2)CC(C)N(C(c2cncc(Br)c2)=O)C1 N1(C(C(COC)C)=O)CCCC(CC(=O)N(C)CCN2CCCC2)C1 c1(C(=O)NCC2CCC(NC(c3cnco3)=O)C2)nsc2c(Cl)cccc12 c1(OC)ccc(F)cc1C(=O)NC1CC(CCNC(=O)COCCF)C1 CN1C(=O)CN(CC(N2CCC(C)(NC(C34CC5CC3C4C5)=O)C2)=O)C1=O C1(CC)(NC(c2cnc(C)nc2C(C)C)=O)CCCN(C(c2cnc(O)s2)=O)C1 c1(COCC)nc(C(=O)NC2(C)CC(NC(=O)C(C)c3cc[nH]n3)C2)cs1 N1(C(c2c(C)nc(C(C)C)s2)=O)CC(C)CN(C(=O)C(C)(C)C)CC1C C(=O)(C1=CCCSC1)NCC(CCNC(C1(OC)CCCC1)=O)O N1(C(c2c(C)n[nH]c2C)=O)CC2CC(NC(=O)C(N3CCOCC3)C)C1C2 Cc1cc(=NC(=O)C2C3CC2N(C(c2cncc(Br)c2C)=O)C3)[nH][nH]1 n1(CC(=O)N(C(C2CN(C(=O)COC3CC3)C2)C)C)ccc(F)cc1=O C1(C(N2CC(N(C)Cc3cccc(CC)c3)C2)=O)COc2ccccc2O1 c1(C(N2CCCC(Cn3cc(C4CCN(C)C4)nn3)C2)=O)cnc(Cl)c(Cl)c1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCCC(CCNC(c2c(C)ccs2)=O)CC1 C1(C)(C(N2CC(NC(C=Cc3cccc(C)c3)=O)C2)=O)CC2(C1)CC(F)(F)C2 C1(C(N(CC(CNC(CC2N(C(C)=O)CCC2)=O)C)C)=O)CCC(=C(F)F)CC1 N1(C(C=CC=CC)=O)CC(NC(=O)CCc2ccccc2C)CC(C)(C)C1 CC1(C)CC(CNC(c2ncc[nH]c2=O)=O)CN(C(c2cc(N)cnc2Cl)=O)C1 C12(CNC(CCC#CC)=O)CCC1CN(C(c1ccc(N(C)C)cc1F)=O)C2 c1(NC(C)=O)ccc2nc(-c3ccccc3)oc2c1.C12(F)CC(C1)NC2=O CC(C)CC(CNC(C1CC2CCCC2C1)=O)C(=O)N(c1cccc(C#N)c1)C c1(C(=O)NCC2CC(F)(CNC(C(C=C)(C)O)=O)C2)cc(O)nc(OC)n1 C1(OC)CC(O)CN(C(=O)CC2C3CCC(C3)N2C(C2CNC(=O)O2)=O)C1 N1(C(c2ccc(C(C)=O)c(F)c2)=O)CC(O)C(O)C1(C)C C1(C(=O)NCc2c(C(N3C(C)(COC)CC3)=O)n[nH]c2)COCC(C)O1 C1(C(=O)NC2C(C)(C)C2C(=O)NCCCCC(N)=O)CC2CCC2C1 c1(C(=O)Nc2cc(C(=O)NC(C)C#N)n(C)c2)c2c(nn1C)CCC2 C1(NC(COCc2onc(C)n2)=O)CCC(C)(CNC(c2ncn(C)c2C)=O)C1 c1(CC)[nH]nc(C(=O)NCC(CC)(CC)NC(C2C=CCS2)=O)c1C C12(NC(c3cscc3F)=O)CC(NC(C34CC(CC(F)(F)F)(C3)C4)=O)(C1)C2 C(=O)(C1=CCSC1)N1CC(CC(=O)NCCCSCCO)C1 c1(NCCS(CC)(=O)=O)nc(=NCC(CO)C2CC2)[nH]c2cc(C)ccc12 CCCCC(F)C(=O)N1CCC2C(C(=O)NCCC(O)C(F)F)C2C1 c1(C(=O)NC2CC3(CC(NC(=O)OC(C)(C)C)C3)C2)ccc2c(O)ncnc2c1 CC1CN(C(=O)C(C)N(C)C)CC1(C)CNC(c1cn(C)nc1-c1ccoc1)=O c1(C(N2CCC(NC(C(CC)NC(C)=O)=O)C(F)C2)=O)c(OC)ncc(Cl)c1C c1(CC(N2CC(NC(CC)=O)(COC)C2)=O)cc(CC)nn1C C12(C(=O)NCCCN(CC)CC)CCC(CN(C(=O)C(CO)NC(N)=O)C1)C2 C1(CC(=O)NC2(C(=O)OCC)CCCCC2)CCCCN(C(=O)CSC)C1 Cc1ccc(F)c(OCC(=O)N(C2CCN(C(=O)CSCC(N)=O)CC2)C)c1 C1(C(=O)NCC(=C)F)CC2(CCC2)CN1C(=O)CCCF c1(C2C(C(=O)NCC3CCN(C(C=CC(C)C)=O)CC3)C2)c(Cl)cccc1Cl N1(C(COCC=C)=O)CCCC2(CCCN2C(C2CC2c2cccc(O)c2)=O)C1 C(CCC(=O)NC1CC(F)(CF)C1)N(C(=O)OC)C.C12CCCC1C(=O)N2 N1(C(C(c2ccc(COC)cc2)=O)=O)C2CCC1(C1CCCOC1)CC2 CC1CCc2ncc(C(=O)NCCCN(CCO)C(C3(C)CCC3)=O)n2C1 C12CCN(CC1)CCN1CC(O)(C1)C2C.c1(C(=O)NS(C)(=O)=O)cccs1 C(C1CCCn2ccnc21)NC(C1(c2nnc(C)s2)CC1)=O N1(C(=O)NC(c2nc(Cc3ccc(F)cc3)cs2)C)CCC12CCN(C)C2 N1(C(c2c(C)ncn2O)=O)C2CCC1CC(NC(C1CCCN(C(N)=O)C1)=O)C2 N1(C(C(CC(C)C)ONC(c2c(C)cc(CC)o2)=O)=O)CCC(O)C(C)(O)C1 c1(CNCC2(OC)COC2)cc(S(N)(=O)=O)c[nH]1 N1(C(CC2(C(=O)NC3(OC(C)C)CCC3)CC2)=O)CCN(CCO)CC1 CCC(C(=O)NCc1ccc(CNC(C2CCCS2(=O)=O)=O)cc1F)C(C)(F)F C(C)(C(=O)N(C(C)CNC(C1CCCS1)=O)C)SCCCC N1(C(C=C2CCC(C)CC2)=O)CCN(C(=O)CCC2CC2)C(C(C)(C)C)C1 c1(C(=O)NCC(C)CNC(c2cc(C(F)F)n(C)n2)=O)cc(F)cc(Br)c1 C1(CNC(COCc2onc(C)n2)=O)CN(C(c2cccs2)=O)CC12CCC2 Cc1ccc(C(N2CC(NC(C3CC4(C3)CC4F)=O)C(C)C2)=O)c(C)n1 C1(C2(O)CN(C(=O)N(C)CCOC)C2)(CNC(c2cc(CC)on2)=O)CC1 C1(C(=O)NC(C(=O)NC2(CSC)CCC2)CC2CCC2)C=CC=CC=C1 N1(CCCNc2nn(CC)c(C)c2)CC(C)CC(C)C1 C(=O)(CC1=CCCC1)NCC1(F)CCC(NC(C(C)(F)F)=O)C1 c1(C(=O)NC(CC(C)C)CNC(c2cnc(N(C)C)nc2)=O)nn(C)c(Cl)c1Cl c1(OC)ccccc1C1CC(OC(C2(Br)CC2)=O)C1 CC1COCC(CNC(=O)CC(C)NC(C2CC2C(C)(F)F)=O)O1 C12(C(N3C(CC)(CC)CC3)=O)CCCC1CCN2C(=O)C(C1CCCCC1)C c1(OC)cc(C(=O)NC(CC2CCC2)C(=O)NCc2nc(C3CC3)n[nH]2)[nH]n1 N1(C(CNC(CC)=O)=O)CCC(COC)(NC(=O)CCc2ccc(C)o2)C1 Cc1ccc(S(=O)(=O)CC(C)Nc2nnnn2Cc2cccc3c2ncn3C)cc1 CCC(CC)(C(=O)N1CCCC1CN(C(=O)C(C)S(N)(=O)=O)C1CC1)C(C)C CC(C)CC(C)C(=O)N1CCC(CC(N2CC(O)C(O)C2)=O)C1(C)C C1(C(N2C(C)CN(C(COCCC#C)=O)C(C)C2)=O)CC(C)(C)CC(C)(C)C1 C1(CCNC(Cc2c(C)scc2)=O)CN(C(c2ccncc2N)=O)CC(C)O1 Cc1cc(C)c(C(N2CCCC(CNC(=O)C(C)Cn3ccnc3)C2)=O)c(=O)o1 C1(CNC(C2CN(C(c3cc(OC)n(C)n3)=O)CC2C)=O)COCC(=O)N1C N1(C(CCC(=C)Cl)=O)C2CCC(C2)C1C(=O)NCC(C)CO c12cn(cn1)CCCNC2=O.C1(C(C)(C)O)(C(CC#CC)=O)CCC1 N1(C(=O)Cc2c[nH]nc2O)CC(NC(C2COCC2C(F)F)=O)C2(CC2)C1 C1(N(C(CC=CC)=O)CCC)CCCN(C(c2cc(N3CCCC3)ncn2)=O)C1 N1(C(C(CCNC(c2ccc(C)nc2)=O)O)=O)CCN(C)CC1CCO C(CCC(C)(C)NC(C1(C)CC1F)=O)NC(COC1(C)CCCC1)=O N1(C(C2CCC(C)O2)=O)CC2(CCN(C(c3ccc(CN=[N+]=[N-])cc3)=O)CC2)C1 N1(C(C2N(CCCC)CCOC2)=O)CC2(CCN2C(=O)CCC2CCCO2)C1 C1(CNC(CC(C=C)C)=O)C2CCC(C2)N1C(c1cccc(C2(C)CC2)c1)=O c1(C(=O)OC)ccc(S(=O)(=O)NC2CC3CCC(C2)N3C)nc1 CCC(C)C(CN=c1[nH]c(=NC2CCS(=O)(=O)C2)[nH]c2cccnc12)OC C1(C(N(C(C(=O)NC2C(C(=O)OC)CC2)C2CC2)C)=O)CC12CCOC2 c1(N(C2CC3CC2CC3N)C(c2c(Br)c(C)n(C)n2)=O)ccc2ncnc(O)c2c1 S(=O)(=O)(c1ccccc1)NCCC(=O)NC1CCN(C(CN(C)C)=O)C12CC2 c1cnc2ccnn2c1.C1(C(=O)NC2CC(NC(=O)C[SH2]C)C2)(CO)CCCC1 CC(O)C(F)(F)C(=O)N(CCCNC(=O)Cc1cc(Cl)cs1)CC1CCCC1 Cc1cc(C(=O)NC2CC2NC(=O)CCOc2c(F)cccc2Cl)c(F)cc1Cl CCC(CC)CC(C(=O)NCC)N1CCCCC1Cc1cccc2ccccc12 c1(C(=O)NC(C(=O)N(C(C=C)C2CC2)C)C2CCOC2)sncc1C CC(C)CC(CNC(=O)C(CC#N)c1ccccc1)NC(=O)CCCC1CCC1 C(C)(CO)(C(=O)NCCCN1CCC(NC(=O)COC2CC3C=CC2O3)C1)OC C1(C(NOCc2cn(CCC)nc2)=O)CC(C)(C)CCN1C(=O)CCCF c1(CC)cccc(C)c1NC(=O)C(N1CCNC(=O)CC1)C(C)C1CCOC1 N1(C(C)(C)C)CC(C(N2CCCCC2CNC(=O)CCCCF)=O)CC1=O N1(C(CCCOCCC)=O)CCN(C(c2ccc(CCF)cc2)=O)C(C)C1C N1(C(C23CC(NC(=O)Cc4nncs4)(C2)C3)=O)CCCC(CN2CCC2)C1 CCC(N=c1[nH]c(Cl)nc2cc(C)sc12)C(C)(C)C(=O)OC(C)(C)C c1(COC)cccc(OC)c1OCC(C(=O)NCCCSC)NC(N)=O S(=O)(=O)(c1ccc(C#N)c(NC2CC(C(F)(F)F)C2)c1)N1C(CC)CCCC1 c1(CCC(=O)N(CC(C)NC(C)=O)CC)noc2ncc(C(=O)OC)cc12 C1(NC(C(C)OCC)=O)CCCCN(C(c2ccc(C#N)[nH]2)=O)CC1 c1(N2CC(NC(=O)CSc3ccccn3)CC(C)(C)C2)ncnc2[nH]c(Cl)cc12 Cc1ncc(C(N2CCC(CN(C(c3ccsc3Cl)=O)C3CC3)CC2)=O)n1C c1(C(N2CCC(NC(C(CCC)N(C)C)=O)C(O)C2)=O)nnn2c1C(=O)NCC2 C1(NC(c2cnco2)=O)CCN(C(C2CC2c2cccc(Br)c2)=O)CC1 CC1(C)CN(C(C2(C)CCCO2)=O)CC1CNC(c1ccnc(CO)c1)=O Cc1ccc(C=CC(=O)NCC=CCC(=O)NC2(C(C)(F)F)CC2)cc1 O=S(=O)(C1=Cc2ccccc2OCC1)N(c1ncccn1)CC1CC12CCNCC2 C#Cc1c[nH]nc1C(N1CCN(C2COCC2NC(C2(O)CC2(C)C)=O)CC1)=O C(=O)(C1CCc2c[nH]nc21)N1CC(CC)(NC(C2CC(C)(OC)C2(C)C)=O)C1 C1(NC(CN(C(C)=O)C)=O)CN(C(C2COC(C)(C)C2)=O)CC2(CC2)C1 C1(NC(C(CCC)NC(=O)CCCN(C)C(C)C)=O)CCCCC12CC2 C(CC(F)(F)CO)NC(C(C)CN(C)C(c1cnn(C)c1Cl)=O)=O N1(C(CNC(=O)OC)=O)CCN(C(C2CC3(CCC3)CO2)=O)CC1C C1(C(=O)N(CC(C)N(C)C(C2CC(n3cnnc3)C2)=O)C2CC2)CCC(C)(O)CC1 c1(C(=O)NC2CCN(C(=O)CN3CC(=O)NC3=O)CC2)cncc2nc(O)[nH]c12 CC1(C(N2CCC(F)(C(N3CCC(CO)C3)=O)C2)=O)CCC2CC2C1 C1(CC(N2CCCC(N(C(C(C(C)C)O)=O)C)C2)=O)CCC2(CC1)OCCO2 c1(CC)cc(C(=O)NC2CCCC2NC(=O)CC2CCCCO2)ccc1O Cc1cc(F)c(C(=O)NC2CC2C(N2CCOCC2CO)=O)c(Br)c1 Cc1cccc(CC(N2CC(NC(=O)C=CC3CCCC3)C(C(F)F)C2)=O)c1 c1(C(=O)NC(C2CCC(CN3CCCC3)CC2)C2CC2)c(I)ccnc1F N1(C2CCN(C(=O)COC(F)F)C2)CCN(C(c2n[nH]c(CO)c2F)=O)CC1=O c1(C(=O)NCC2(O)CN(C(C(CN(C)C)O)=O)C2)ccc(O)cc1C(F)F C12(C(N3C(C(=O)OC)CC3C)=O)CC(CN(C(=O)CCC3CCCOC3)C1)C2 c1(C(N2CC(CCNC(C3CC4C=CC3C4)=O)C2)=O)ncc(Cl)cc1Cl c1(C(N(CCCN(C(=O)C(O)C2CC2)C)C)=O)ccc(Cl)c(O)c1N C1(C(N2C(C)CC(OC)C2)=O)CC2(CCN1C(C1CC3C=CC1O3)=O)CC2 Cc1[nH]nc(C(=O)NCc2nc(CNC(C3C4CNC(=O)C34)=O)cs2)c1O c1(CN=C(NC(c2cccc(C#N)c2)C#C)NCC(F)F)ccc(Br)cc1C#N C(=O)(C1CC(=O)Nc2ccccc21)N1CCN(C(CS(C)(=O)=O)=O)CC1CCO Cc1cnc(-c2cn(CC3CCCN3C(=O)C(F)CN(C)C)nn2)c(C)c1 N1(C(c2cnc(C)[nH]2)=O)CCCC2CN(C(c3cccc(Br)c3F)=O)CCC12 C1(NC(=O)NC(CC)CCO)COCCN(C(C)C=O)C1.C(C)(C)(C)O N1(C(C)=O)CCC(C(N(c2cc(Cl)ccc2F)CC=CC2CCCO2)=O)CC1C C(C(C)(C)C(F)(F)F)NC1(c2n(CCCOC)nnn2)CCC1CC(F)(F)F C1(C(N(CC(C)NC(c2cnc(O)s2)=O)C)=O)C2COCC12 c1(CCNS(C)(=O)=O)nc(-c2ccccc2)nn1C12COC(CF)(C1)C2 C1(C(N(CCC(=O)N(C2CCOC2)CCO)CC#C)=O)CCN(C)C1C c1(CC(=O)NC2CC(OC)CN(C(CC=CCC)=O)C2)c[nH]c2c(F)cccc12 C1(CNC(CCN(CCC)C)=O)CC2COCC2N1C(C1CCCSS1)=O CCC(C)C(O)CC(=O)NCC1(NC(C2(CC)CC(C)(C)C2)=O)CC1 C#Cc1cccc(CC(=O)NCCNC(c2ccc(C(C)=O)cc2)=O)c1 N1(C(CCOC)=O)CCOC2(CCC(NC(=O)C3=CC(C)(C)C3)CC2)C1 C(=O)(C(CCN(C)C)NC(C1CC12CCC2)=O)N(C)Cc1n(CC)ccn1 N1(C(c2cnn3cccc(OC)c32)=O)CCC2CN(C(=O)C=CSC)CCC12 N1(C(C(N2C(CC)CCC2)=O)=O)CC2(CCN(C(C3CN(S(C)(=O)=O)C3)=O)C2)C1 C(=O)(CCC(C)NC(c1ccsc1)=O)NC(C(=O)NC(C)C)C N1(C(C2(C)C(C)(C(=O)OC)CC2)=O)CC2(CC(NC(=O)C(C)N3CCC3)C2)C1 c1(C(=O)NC(c2ccccc2)CCC)c(-c2sccc2C(F)(F)F)cncc1F N1(C(C2(C)CN(C(C=CC(=O)OCC)=O)C2)=O)CCCC(F)(F)C1 C(=O)(C1=Cc2ccccc2N(C(=O)OC(C)(C)C)C1)N1CC(C)(CC)OCC1 C(=O)(C1CCc2cccc(Cl)c21)N1Cc2c(ccc(NC(c3nc[nH]n3)=O)c2)C1 CCC(F)(F)C(C)(C)NC(C1CN(C(c2ccc(SC)o2)=O)CC12CC2)=O c1(C(=O)NCC(C)CN(C)C(c2ncoc2C2CC2)=O)cnc(O)c(Br)c1 c1(CNC(CN2CCn3c(C)ncc3C2)=O)c(O)nnc2c1COCC2 c1(NC(C23C(NC(C=CC(C)(C)C)=O)C4CC2C3C4)=O)cccc2ccccc12 C1(CNC(C(CCC)C)=O)CC2(C1)CN(C(=O)Cc1ccc(C)nc1)C2 CC1(C(=O)NC2CC(CNC(C3(O)COC3)=O)C2(C)C)CCOCC1 c1(CCN(C(=O)C(C)(F)CF)C)ccc(F)cc1F N1(C(c2c(CCNC(c3occ(C(N)=O)c3)=O)n[nH]c2)=O)CCC(O)(C(F)F)C1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nnc(=O)[nH]2)ccccc1[N+](=O)[O-] Cc1ccc(C(=O)NC(C)CCN(C)C(C2C=CCS2)=O)s1 C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1CCC(CNC(Cc2c(C)ccs2)=O)C1 C1(C#N)(C(=O)NC2C(C)(C)C(CNC(c3ccc(NC)cc3)=O)C2)CCCCC1 N1(C(C(Cc2ccco2)OC)=O)CC2(CC2)CC1C(=O)NCCC1CCN(C)C1 c1(C(=O)NCCC2CCN(C(=O)CCOC3COC3)C2)ccc2ocnc2n1 N1(C(c2c(C)nsc2N)=O)CC=C(CC(=O)Nc2cnn(CC3CC3)c2)CC1 Cc1cnn(C)c1CC(=O)NC(C)CCCNC(C1CC1C(F)(F)F)=O c1(C(=O)NC(C(C)NC(=O)CCn2ccnc2)(C)C)cc(=O)n(C)cn1 N1(C(c2ccc(C)c(N)c2)=O)C(CNC(c2cccn2C)=O)CC2COCC12 c1(CC(=O)NCCOCCNC(C(F)=C(C)C)=O)c[nH]c2cc(F)ccc12 N1(CC(=O)NC)CC(NC(c2cn(-c3ccccc3)nn2)=O)C(C)(C)C1 c1(C(N2CCC(C(C)NC(c3ccsn3)=O)CC2)=O)cc2cnccc2[nH]1 CC(c1ccsc1)=CC(=O)N(CCCNC(C1(C#N)CC1C)=O)CCO N1(C(c2csc(C)c2C)=O)CCCC(N(C(=O)C2=CCCCC2)CC2CC2)CC1 N1(C(C(C)OC2CCCC2)=O)CCC2(COC(CNC(C3(O)CCC3)=O)C2)C1 CC1(C(=O)NC2CCCC(NC(=O)COCc3ccccc3)C2)CNC(=O)C1 c1(C(=O)NCC(CCNC(C2CC(C)=C(C)CC2)=O)O)cc(F)cc([N+](=O)[O-])c1 c1(CC)cc(CCCN2CCCC(NC(=O)CC3CC(NC)C3)C2)ccc1C C(=O)(C1=CCCCC1)N1CC=C(CNC(c2ccc(CNC(C)=O)o2)=O)C1 CN1CCCC(CC(=O)NC2CC(C(=O)N(C)CC3(C#N)CC3)C2(C)C)C1 N1(C(c2ncc(CC)s2)=O)CCN(C(=O)CN2CCSCC2)CC(CO)C1 Cc1nn(C)cc1C(=O)NC1CC(F)(CNC(c2ccnn2C)=O)C1 C(C(CNC(C1NC(=O)OC1(C)C)=O)S(C)(=O)=O)NC(c1n(C)cnc1)=O C#Cc1cccc(C(N2CCC(CONC(C3CC(OC(C)(C)C)C3)=O)C2)=O)c1 CC1CC(C(=O)N(C2CCN(CC3CC3)C2)C)CN(C(=O)C=Cc2nccs2)C1 C(C(O)CNC(c1cccs1)=O)N(C(=O)C=CCOC(C)(C)C)C Cc1cc(C)oc1CNC(=O)COCCNC(=O)CSc1cccnc1 C=Cc1ccc(C(N2CC(CNC(=O)C(c3ccc(F)c(Cl)c3)(C)C)C2)=O)cc1 N1(C(COCCCC)=O)CC2(CC(NC(C3CCC(O)CN3C)=O)CO2)C1 C12(CNC(C(C)CF)=O)CCCCC1N(C(c1ccc(CCF)cc1)=O)CCC2 c1(C(=O)NC(C2N(C(CC(CC)C3CCC3)=O)CCC2)C)cnc(O)c(F)c1 Cc1cc2[nH]c(C(N3CCCC(NC(c4coc(Br)c4)=O)C3C)=O)cc2o1 C12(C(=O)NC3C(C)(C)C3c3ccc(F)cn3)CCOC(c3cccs3)(C1)C2 c1(OC(CC2(C(C)NC(C(=O)NC)C3CC3)CC2)=O)ccc(CO)nc1 c1(C(N2C(C(N3C(C)C(O)CCC3)=O)CC(F)(F)C2)=O)cc2cc[nH]c2cc1F Cc1c(CN2CCCCC2c2ccc(Br)cc2)cnn1C(C)C C(=O)(CC(C)(C)NC(c1cc(OC)ns1)=O)NC(C#C)C C1(C(=O)NCC2(C)CC(O)C2)CN(C(=O)CC2CCCCC2)CC12CC2 C1(CC)CN2CC1C2=O.c1(CC(=O)NCC2(CO)CC2)cnccn1 CCC(Cc1ccc(N)cc1)C(=O)N1CC(NC(=O)CSc2nc[nH]n2)C2CC2C1 c1(OC)ccc(C(CNC(=O)C(C)(C)OC)NC(=O)CC(C)SC)cc1 CC1(CCC(=O)NCC2(CO)CC23CCC3)CCCN1C(=O)C=CC(F)F C1(N(C(=O)CC2(O)CCC2)C)CN(C(C2(C)CC(F)(F)C2)=O)CC1O c1(SC)cn(C)nc1C(=O)NCC(C1CCN(C(c2ns[nH]c2=O)=O)CC1)(C)C CC1(N2CCC2)CN(CCNC(=O)CCNS(C)(=O)=O)C1 c1(C(=O)NC(CN(C(C(F)=CC)=O)CC)C)cc2c(C)cc(C)cc2[nH]1 Cc1nc(N2CCN(C(c3nccnc3N)=O)CC2C(C)C)cc(C(C)C)n1 Cc1nn(C)c2cc(NC(C3CC34CCN(C(=O)Cn3ccnn3)C4)=O)ccc12 c1(CC)cc(C(=O)N(CCCNC(C2CN(C)CCO2)=O)C2CC2)n(C)n1 c1(C(N2CC(C(C)NC(CCC(=O)NCC)=O)OCC2)=O)c(C)ccnc1C N1(C(CC2(NC(=O)Cc3ccccn3)CC2)=O)CCN2CCC1C2 CC1(CN=c2ccnc[nH]2)CCCN(C(C2(O)CCC2)=O)C1 N1(C(c2c(C(C)NC(c3cc(=O)cc[nH]3)=O)noc2)=O)CCC(F)(F)C(O)C1 c1(C(N(C2CCN(C(CC3CCC(=O)O3)=O)C2)CCO)=O)ncncc1Cl C1(NC(CC=C)=O)CCCC1NC(=O)C(F)(F)c1csc(C)c1 CC1C(NC(=O)CCCCO)CCCN1C(C1(F)CCCC1)=O c1(C(=O)NC2CCC(CCNC(COC)=O)C2)nn2c(c1C)CCCC2 C(=O)(CC(C)CC(C)C)NC1C(C(=O)NCCCCCCCC)CCC1 C(=O)(CC(c1ccccc1)N(C)C)NCC(C)NC(c1csc(C(C)(F)F)n1)=O N1(C(C(=O)NC(C)C)=O)CC(CO)C2(C1)CN(C(=O)C(O)C1CCCC1)C2 Cc1cn2nc(C(=O)NCC3CN(C(=O)C(C)(C)CF)CC34CC4)cc(C)c2n1 c1(C(N2CCCC(NC(c3cncc(Cl)c3)=O)C2)=O)ccc2cccc(Cl)c2n1 c1(C(C)C)nocc1C(=O)NC1CC1CC(=O)NCCc1ocnc1CC1CC1 C1(CNC(CCC=C)=O)CCC(C)(C)CN1C(=O)CSCC(F)(F)F Cc1cc(C(=O)NC2CC(CNC(=O)C(c3ccc(Cl)c(Cl)c3)O)C2)ncc1Cl C(CC(C(=O)NCC=CCNC(C1CC1c1cccc(COC)c1)=O)OC)OC Nc1ccc(F)cc1C(=O)NCC1CC(NC(=O)CC2CCCCC(=O)N2)C1 c1(N(C)Cc2cccnc2Br)ccc(S(=O)(=O)N(C)Cc2ncnn2C)cc1F Cc1cncc(C=CC(=O)NCC2(C)CN(C(=O)CC3CCSCC3)CC2C)c1 C12(NC(C3CC(NC(c4cnc(COC)s4)=O)C3)=O)CCC(CC1)C2 C1(NC(c2cccc(N(C)C)n2)=O)CN(C(C2COC(=O)N2)=O)C2(CCC2)C1 c1(C(c2nnnn2CCC2(C)CC2)NCC(C)CO)ccc(Cl)c(F)c1F N1(C(C(C)=C(C)C)=O)CCC2C(CCCN2C(c2snc(O)c2Cl)=O)C1 C(=O)(C(CCCOC)NC(=O)C=C=C(C)C)N(C(C#C)C1CC1)C N1(C(c2cnn(CC)c2C)=O)CCC2CC1CN(C(=O)CCN1CCOCC1)C2 c1(C(=O)OC)ccc(S(=O)(=O)N2CC(F)(C(=O)Nc3ccc(Cl)nc3Cl)C2)n1C CN1CCN(C(C2CCCSS2)=O)CC1CNC(=O)CC1CC2CC2C1 Cc1nc(CC(C)C)oc1C(N1CC(CNC(C2CC(F)C2)=O)C(C)C1)=O C1(C(=O)NCC2CCN(C(C(CC)CC)=O)C(C)C2)C2CCC(C2)C1(C)C c1(C(=O)NCC(CC=C)NC(=O)C(N2CCCCC2=O)C)cncc(C)c1 N1(C(c2cccc(C(C)=O)c2)=O)CCC2(CCCN(C(c3cnoc3C)=O)C2)C1 C(C(C)(C)C(C)(C)O)N(C(CN(C)C)C(=O)NC1CC1)C(C=C(C)C(C)C)=O c1(C(=O)NCC2C(NC(c3c(F)ccc(C)c3)=O)CC2)cccc2c1NCC2 c1(NCCCn2c(C)nnc2)ccc(S(=O)(=O)N2CC3CC=CC2C3)cc1Br C1(C)(C(=O)Nc2nc(C)c(C(F)F)cc2)CC(C2CC2)=NO1 Cc1ccc2oc(C(N3CCCSCC3C)C(=O)NCCC3(C)CC3)cc2n1 C(=O)(C1CCc2c[nH]nc21)N(C(CNC(=O)CC(C)(C)C(F)(F)F)CC(F)(F)F)C CON(CCO)C(=O)C1CC(NC(C2(F)CC=CCC2)=O)CCO1 c1(C(N2CC3N(C(CCCC=C)=O)CC(C3)C2)=O)c(C)c(C)nn(C)c1=O N1(C(CN(C2CC2)CC)=O)CCc2ccccc2C1CNC(=O)CC1CC1C C1(NC(CC(=O)NCC)=O)CN(C(=O)Cc2ccoc2)CC1N=[N+]=[N-] C1(C(N2CC(F)(CNC(CC3(C(=O)OC)CC3)=O)C2)=O)CC12CCSCC2 N1(C(C)=O)CSCC1C(N1CCC(C(C)N(C(=O)C(c2cccnc2)C)CC)C1)=O C1(C2(O)CCN(C(C3(C)CC3(F)Cl)=O)CC2)(NC(Cn2c(C)nc(C)n2)=O)CC1 N1(C(C2CCCCCC2)C)CCC2(CN(C(c3occc3C3CC3)=O)CCO2)C1 C1(C(=O)NC2C(NC(C(CC)N3CCCC3=O)=O)C2)CC2CCC(C1)O2 Cc1coc(C(N2CCC(N(C)C(c3cncc(CO)c3)=O)C2)=O)c1C c1(C(COCCN(CCCNC(=O)CCOC)CC)(F)F)ccccc1 C(=O)(C(O)C(C)(C)C)NC1(C)CN(C(Cc2cccc(OC)c2)=O)C1 C1(C(N2CCCC2CN(C)C(C2(C)CNC(=O)C2)=O)=O)(OC)CCCCCCC1 C1(C(N(CCN(C)C(c2c(C(F)(F)F)cnn2C)=O)C)=O)Cc2ccccc2N1 N1(C(c2c(OC)cc(OC3CC3)cc2)=O)CCOCC(C)(CNC(=O)CO)C1 CC1COCCC1N(C)C(C1(O)CC(CNC(=O)CN(C2CCC2)C)C1)=O C1(CN(C(=O)C(C)CCOC)CC)CCN(C(=O)CCc2cc(C)nn2C)CC1 Cc1cc(C2(C(=O)NC3(CCNC(=O)CNS(=O)(=O)C4CC4)CCC3)CC2)no1 C(=O)(C1COc2ccc(Cl)cc21)N(C)CC1(O)CCN(C(CCNC(C)=O)=O)C1 c1(C(=O)NCCC2CC(NC(CSC(C)C)=O)C2)ccc2c(c1)CCCS2 N1(C(c2cc(C)c(C)s2)=O)CC(C)(C)CC1CNC(c1cc(C(F)F)cs1)=O c1(CC(=O)NCC(C)CN(C(=O)CCCF)C)cc(O)nnc1O C1(C(=O)NCCCN(C(=O)C(F)(F)c2ccnn2C)C(C)C)CCC2CC12 C1(C(=O)NCCC(C)NC(=O)CNC(=O)C2CC2)CCC(C(N)=O)O1.c1(S)ccccc1 C1(C(NS(=O)(=O)NCC(F)(F)F)=O)CCCN(CCSC2CC2)C1 C1(C(N2C(CCCC)CN(C(C3CC3C)=O)CC2)=O)CC12CCC(C)(C)CC2 Cc1cc(C(N2CC=C(CNC(c3cc(Cl)cnc3C)=O)CC2)=O)cn(C)c1=O C1(C(=O)NCCC2CN(C(c3n(C)c(O)nc3)=O)C2)CC2CCC1C21CC1 N1(C(c2cn(CCC)nc2)=O)CC2(CCC2)CC1CNC(c1c(C)nsc1C)=O n1(CCOC)nc(-c2cncnc2)nc1C1CNC(=O)C1 O=S(=O)(c1cccnc1N1CCC(O)C(F)C1)NCc1cn(C2CCC2)nn1 N1(C(CC(CC)SC)=O)CC2CCCC2(C(=O)NCc2ccc(O)cc2F)C1 Cc1ccc(C(N2CC(NC(C3(C)CC(C)(C)C3)=O)C(O)C2)=O)nc1 CC1(C(N2CCCC(F)(CNC(C3(Cl)CC34CCC4)=O)C2)=O)CC2CCC1O2 C1(O)(CN(C(=O)COCc2ccnn2C)C)CCCN(C(C2(C)C=CCC2)=O)C1 CN1CC(NC(c2c[nH]nc2CNC(=O)Cc2ccc(O)c(F)c2)=O)C(C)(C)C1 C(C1CN(C(c2cnc(CC)nc2)=O)CC1C(N1CCC(NC(C)=O)C1)=O)=CC C12(C(N3CCCC(C)(CO)C3)=O)COCC1CN(Cc1cccc(Cl)c1)C2 c1(CNC2CC(C(N3CCC(C)C3)=O)C2)c[nH]c2c([N+](=O)[O-])cccc12 C1(NC(CC2CCC(C)C2)=O)CC2(C1)CC1(CC(NC(=O)C(c3ccccc3)=O)C1)C2 c1(C(=O)NCC2CC(NC(c3ncc(SC)s3)=O)C2)ccc(OC(C)C)nc1 N1(C(C(CNC(C(C)(C)OC)=O)N(C)C)=O)CCc2ccsc2C1 Cc1ccccc1C1CN(C(C2(N)C=CCC2)=O)CCO1 N1(C(C2CC(=C)C2)=O)CC2C(NC(=O)COCC(=C)C)C2C1 C1(C(=O)NC2C=CCN(C(Cc3c(C)cccc3)=O)C2)CCC2(CC1)CC2(F)F n1(CC)c(C)cc(C(=O)NC(C)C(CO)NC(c2ccc(N(C)C)cc2)=O)c1C N1(C(C(C)(N(C(CCCOCC)=O)C)C2CC2)=O)CCC(CO)C(C)C1 O=C(CCCCO)NCCCCCCNC(=O)CNC(C1COCCOC1)=O CC(C)C(O)C(F)(F)C(=O)N1CCCC(N(CCF)C(c2cccn2C)=O)C1 c1(C(=O)NC2CN(C(Cc3nc(C)[nH]n3)=O)C(C)C2)nc(O)nc(O)c1F Cc1cc(C(=O)NC2CN(Cc3c(O)cc(F)cc3F)CC2(F)F)cc(C)c1F c1(C(N2CC(NC(CCCCOC)=O)C(OC)C2)=O)cnc2ccccc2c1 c1(CC)onc(C(=O)NCC23CC(NC(c4cnc(C5CC5)s4)=O)(C2)C3)c1C C(N=c1[nH]cnc(O)c1Br)C1CC(NC(c2c(CC)n[nH]c2)=O)C1 CC1CC(C)C(C(=O)NCC2CC3(CC(NC(c4ncn(C)n4)=O)C3)C2)CC1C S(=O)(=O)(c1ccc(C(C)C)cn1)NCCCC C#CCC(C(=O)NC(CC)CO)NC(=O)C=Cc1nccs1 C12(CNC(C3(C#C)CC3)=O)CCCC1N(C(=O)C(COC)CC)CC2 c1(C(=O)NC2C=CCN(C(c3cccc(C)c3N)=O)C2)ncccc1S(C)(=O)=O CCC(COC)C(=O)N1CCC(CN(C(=O)CCCCSC(F)(F)F)C)CC1 N1(C(C(c2cn(C)nn2)NC(CN(CCC)C)=O)=O)CC2(CCC(O)CC2)C1 C1(CNC(C(C)SCC)=O)CCN(C(C2CCN(OCC)CC2)=O)C12CCC2 C#CCC(C)(C(=O)NC12CCOC(C)(C1)C2)NC(=O)COCCF c1(C(=O)NC(C(C)NC(CN(CCC)C)=O)C)c(OC)cc(OC)cc1CC C(=O)(CC(C)(C)C=C)NC(CC(=O)NC(C#C)C1CC1)C CC1(C(=O)NC2C3CC4C(C3)C24C(=O)NCCOCC2CC2)CC2CCC1O2 N1(C(c2ccc(CC)[nH]2)=O)CC2CCC1CC2NC(=O)C(c1cn(C)nc1C)C CCC(CC)CC(=O)N1CC(NC(c2csc(-c3nc[nH]n3)n2)=O)C(F)C1 c1(CC2C(=O)CC(CCc3ccccc3)N2)ccc(Cl)cc1.CO Cc1cnc(C(=O)NCC(C)(C)CCNC(c2ccc(C(N)=O)cn2)=O)c(F)c1 c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)C)oc2c(c1C)C(=O)CCC2 CC(CC1CCC1)C(=O)N(C(c1nnnn1C1CC1)C1CCCCC1)C1CC1 N1(C(c2csc(C)c2C)=O)CCC2CN(C(=O)C(C)(C)n3cccn3)CCC2C1 C=CCC(CC(=O)NCC(O)CC(=O)OC)NC(C1(C)CC(C)=NO1)=O c1(C(=O)OC2CC(CCC3CC(F)(COC)C3)C2)ccc(Cl)cn1 N1(c2c(C#N)c(N3CCOC(CO)CC3)ncn2)CCn2ncc(Br)c2C1 c1(N(CC)CC2CCN(C(=O)C3=NOC(C)C3)CC2)ncnc2[nH]ccc12 C1(N2CCOCC2)(C(=O)NCCCN(C(C2CC2F)=O)C2CC2)CCCC1 N1(C(C2N=C(C)SC2)=O)CCC(C2(NC(=O)CC3=NNC(=O)C3)CC2)C1 Cc1cn2c(CCC(N3CC(NC(=O)Cc4ccccc4)C(O)C3)=O)csc2n1 C(=O)(C1COc2cc(C)c(C)cc21)N1C(CCNC(CCCOC)=O)CCC1 N1(C(C(C=C)O)=O)CC(N=[N+]=[N-])CC1C(=O)NCCC1CC1C N1(C(C(C2CN(C(C3CC3(C)C(F)F)=O)C2)O)=O)CC2C(C1)C2(F)F C1(C(N2CC(CCC)OCC2)=O)CNC(=O)CN1C(c1cc(C)sn1)=O CCCC(CCC)C(C)(c1nnnn1CC1CC1)NCCCCn1ccnc1 c1(NC(C2N(C(CCC#C)=O)CC2)=O)ccc(Br)nc1C(=O)OC C(N=c1nc(C)c(Br)c[nH]1)C1(NC(C=C(C)Cl)=O)CCCCC1C c1coc(CNCCCSCC2CC=CC2)c1 C(=O)(C(C)C(C)(F)F)N1CC(CC(C)CNC(=O)C=Cc2ccc(Cl)s2)C1 N1(C(C#CCNC(c2c(CCC)nco2)=O)=O)CCCC12CCNC2=O c1(C(=O)NC2CC(CNC(C3(N4CCCC4)CC3)=O)C2)cn(C2COC2)nn1 Cc1ccccc1CC(=O)NC1CN(C(=O)C(C)C#N)CC1O N1(C(c2ccc(C(=O)OC)nc2)=O)C(C)C2CC1C2NC(=O)Cc1cc(C)on1 Cn1nccc(C(=O)NCCC2(NC(c3ocnc3CC3CC3)=O)CC2)c1=O c1(C(=O)NCC(C(C)C)NC(=O)C(c2cccc(Cl)c2)C)nn(C)cc1[N+](=O)[O-] n1(CC)ccc(C(N2CC(NC(C3NC(=O)OC3C)=O)CC2(C)C)=O)cc1=O N1(C(CSc2nc(-c3cc(C)c(Br)cc3)oc2)=O)CCCC(O)C(F)CC1 C1(NC(C(=C)F)=O)CCC2(C1)CN(C(c1ccc(O)c(C(F)(F)F)c1)=O)C2 c1(C(=O)O)ncccc1CN(C)Cc1ccccc1 C1(NC(C(n2ccc(C)n2)C)=O)C=CCN(C(=O)C=CCOC(C)(C)C)C1 C=CCCCCCCC(=O)N1CCOC(C)C1C(=O)NCC(F)(CC)CC C(=O)(C(C)(C)C(F)F)N(CC(CNC(CC1(COC)CC1)=O)C)C N1(C(c2n(C)c(O)nc2)=O)CC(CNC(=O)CCS(C)=O)C(C)(C)C1 C1(CC2(C(CNC(NNc3c(C)nsc3)=O)=O)CCCC2)CCN(c2nccs2)CC1 CC1(O)CON(C(=O)C23CC2CN(C(c2cn4ccccc4n2)=O)C3)C1 N1(C(CN(C(=O)OC)C)=O)CC(CC(=O)N(CCN2CC3CC3C2)C2CC2)CC1C CC1CCN(CC2CC3CNC(C2)C3)CC1C N1(C(C(c2ccc(F)c(Cl)c2)C)=O)CC(NC(c2cccn2C)=O)C(C)(C)C1 c1(C(N2CC(CNC(C3CN(C(C)C)C3)=O)C(C)CC2)=O)cc2cccnn2n1 Cc1c(CNC(C2(CO)CCN(C(C)C)C2)C)[nH]c2c(C)cccc12 Cc1noc(C2CC2)c1C(N1CC(CCNC(c2ccsn2)=O)C(C)C1)=O C1(CCCNC(c2c[nH]c(C(N)=O)c2)=O)CN(C(C2CC=CC2)=O)CCO1 C1(C(N(CCCCC#C)CC)=O)CN(C(C)Cc2ccsc2)CCC1O C1(C(C)C)CN(C(=O)CP(C)(C)=O)CCCN1C(=O)CCN(C)CCO c1(SC)nc(O)nc(C)c1C(N1CC(CC(C)NC(=O)CCC(C)N(C)C)C1)=O CC1(C(=O)NCC=CCNC(=O)Cn2ccc(C(F)(F)F)n2)COCCO1 CC1CN(C(c2ccc(N)cc2Cl)=O)CCC1CNC(=O)C(C)(C)COCCO N(C(=NCCCCl)NCc1nc(C(N)=O)cs1)CC1C(C)C1(F)F c1(C(=O)NCCCN(C)C(c2ccns2)=O)nn(C2CCOCC2)cc1[N+](=O)[O-] c1(C(C)C)ccc(C(=O)NC2(C)CC(NC(C3CC3(C)C)=O)C2)c(O)c1 c1(C(=O)NCC(C)NC(CCCOCC=C)=O)cc2c(F)c(Cl)ccc2[nH]1 CC1(C)CC(CNC(=O)CCC2(C)CC2)N(C(=O)COC(C)(C)C)C1 CC(=O)CCCC(C)C(=O)NCC1CCCN(C(=O)CN2CCCC2)CC1 CCCCC(C(=O)NCC(C)N(C)C(c1nc(C(C)(C)C)no1)=O)C(C)C C=Cc1cnn(C)c1C(=O)NCCCN(C)C(C1CC12CC(O)C2)=O N1(C(Cc2cc(C)sc2)=O)CCN(C)CC1C(=O)NC1CCN(C2CC2)C1=O c1(C(=O)NCC23N(C(CCSCC)=O)CCC2CC3)cc2nc(Cl)ccc2s1 N1(C(c2c(C)nns2)=O)CCN(C(C2CCCC3CCCN23)=O)C2(CCC2)C1 N1(C(C(C)OCC=C)=O)CCCC1C1CCN(C(=O)CNc2ncccn2)C1 C1(NC(=O)CN2CCCC2)CCCCN(C(=O)CC2CCCCC23CC3)C1 C12(CNC(C3C(CNC(c4ccsc4)=O)C3)=O)CCN(CC1)CC2 N1(C(c2c(C)c(O)ccc2)=O)C2CCC1CN(C(=O)C(C)C(F)F)C2 c1(OC)cc(OC)c(C(=O)NCC(O)CNC(=O)CC2CCNC2=O)c(N)c1Cl N1(C(C(C)C)=O)CCC(CCC2CCN(C(=O)CC3CCCCN3)CC2)CC1 c1(C(=O)NC(CC)CN(C)C(c2nncs2)=O)c[nH]nc1-c1ccnn1C N1(C(C(C)(C2CC2)OC)=O)CCN(C(c2cnn3ccsc23)=O)CC1COC c1(OC)c(C(=O)NCC2CCN2C(=O)C(C)N(C)C2CC2)scc1Br C(N=c1cc(NCCc2cccc(Cl)c2)nc[nH]1)C1CCC(C)(C)CC1 c1(CC#N)ccccc1C(=O)NCCN(C(=O)CC1(C)CC1(Cl)Cl)C1CC1 n1(CC(N2C(CNC(CC(C)C)=O)C(C)CCC2)=O)ccc2ccc(F)cc12 C1(C(N(CCOCC=C)C)=O)CC(NC(=O)C(C)n2cnnn2)C(O)C1 CC1(C2CCN(C(=O)CCOC3CN(C(=O)CC4CCSC4)C3)CC2)CC1 CCCC(C)(O)CC(=O)N(C)CC1CCN(C(=O)CCOCC)C1 N1(C(C(C)(C)F)=O)CCc2c(C(=O)Nc3c(O)cccc3Br)csc2C1 C1(CC(=O)NC2(CNC(CCOC(C)C)=O)CC2)COCC(C)O1 N1(C(C(C)N(C(=O)C(C)N(C2CC2)CC)CC)=O)CCN(C2CC2)C(=O)C1 CC1CC(NC(C2(n3cccc3)CCCC2)=O)CCN1C(c1ccc(Cl)cc1)=O C(CCCC(C)(C)NC(=O)CC1CC2C=CC1C2)NC(c1cc(C)nnc1)=O C(=O)(CS(=O)(=O)C(C)C)N1CC(C)C(NC(=O)Cc2ccc3c(c2)CC3)CC1 Cc1ncnc(O)c1CCC(=O)NCC1CN(C(=O)Cc2nncs2)C1 C1(C(C(N2CCC(OC)C2)=O)C)CCN(C(=O)CCNC(=O)OC)CC1 c1(C(N(CCN(C(CC(C)n2cccn2)=O)C)C)=O)ccc(C#N)o1 C1(Cl)(C(N(CCCNC(c2ccc(C(=O)OCC)s2)=O)C)=O)CC12CCC2 c1(CC(=O)NC2CCCC(NC(=O)OCc3ccccc3)C2)ccc(Br)c(Cl)c1F N1(C(c2c(C)cns2)=O)CCN(C(C2CCCCN2C(=O)CC(C)C)=O)CC1 CP(C)(=O)C1CCCC(NCC(c2ccncc2)C2CCC2)C1 C=CC(C)(CC)C(=O)NCC1CC1C(N1CCC(CO)C(O)C1)=O Cn1cc(C(=O)NC2CC2CNC(c2ccc(CCO)cc2)=O)ncc1=O C1(C(=O)NC(C(=O)NC2(C)CC(F)(F)C2)Cn2cncn2)CC12CCCCC2 C1(CNC(C2CC(CC)OCC2)=O)CN(C(C2CC(OC)C2)=O)CCCO1 N1(C(=O)C(Cl)=CCl)CCN(C2CCCN(C(C3(C(F)F)CCC3)=O)C2)CC1 N1(C(c2c(C)oc(C)c2C)=O)CCCCC2(CCN(C(=O)CCC3CC3)C2)C1 C12(C(=O)NCCCN(C(C)C)C(c3sccc3Cl)=O)CCCC1CC2 Cc1cnc(C(=O)NC2CCOC(C3CCN(C(=O)C(Cl)=CCl)CC3)C2)c(C)c1 C1(C(=O)NC(C2CCN(C(CC(C=C)C)=O)CC2)CO)CCn2cncc2C1 c1(C(=O)Nc2cccc(CNC(=O)CC3CCC(O)C3)c2)cnc(O)c(Cl)c1 CCC(C)C(O)CC(=O)NCC1(NC(=O)Cc2cn(C)cn2)CCCC1 c1(CCC(=O)N(C)CC2CCCCN2C(c2ccco2)=O)ccccc1[N+](=O)[O-] c1(NC(C2CC(n3ccnc3)C2)=O)cc(Br)ccc1OC(F)F N1(C(CC2N(C(C(CN(C)C)O)=O)CC2)=O)CCC(F)C(F)C1 Cc1nnc(CC(=O)NC2COCCC2NC(=O)C(c2ccccc2Cl)C)n1C C1(C(=O)NCc2ncn(C)c2)CC(O)CN1C(=O)C(CN(C)C)N(C)C N1(C(C2(C#N)CCSCC2)=O)CCC(C2CC2)(CNC(=O)C(F)(F)C(F)F)C1 c1(OC)ccnc(-c2nc(CC(C)C)n(C(c3cc(Br)cs3)C)n2)c1 C12(C(=O)NCC(CN(C(c3cc(C(C)=O)oc3)=O)C)C)CCCN(CC1)C2 c1(CNC(=O)CC2CCN(C(=O)C(=O)C3CCCC3)C2)ccc(Cl)cn1 c1(OC)cc(NC(=O)C(=O)NC2CC(CSC)CC2O)c(N(C)C)cc1Br c1(C(N2C(CNC(C(C)OCCOCC)=O)CCC2)=O)ccc(C)c2c1CCC2 c1(NC(C2N(C(C3(CC=C)CC3)=O)CCC2)=O)ccc2c(c1)OCO2 C1(C)(NC(c2cnn(CC)c2C)=O)CCCN(C(C2CC2C(C)O)=O)C1 C1(C(=O)NCCC(c2cccs2)N(C)C(c2nc(=N)cc[nH]2)=O)CCCCC(=O)C1 c1(C(=O)Nc2scc(C)n2)cc2c(s1)CCN(C(C1(n3cnnn3)CC1)=O)C2 O=C(CCCC(F)(F)CO)NCC1CC1CNC(c1scc2c1OCCO2)=O C12(NC(CC(C)=CC)c3nnnn3C3(C)CC3)CC3CC(CC(C3)O1)C2.C1=CC=C1 CC1=C(C(=O)N2CC(O)(C(C)NC(C34CC5CC3C4C5)=O)C2)CCC1 C1(C(=O)NCC=C)(CNC(c2ccnc(COC)c2)=O)CCOCC1 CC1(C)CCN(C(=O)CCCn2ccnn2)CC1NC(C1CC(=O)C12CCC2)=O c1(CN2CC(C(=O)NC(c3nccc(CC)c3)=O)OCC2)cc(C)c(Br)cc1F C#Cc1ccc(C(N2CCC(NC(c3ccncc3F)=O)C(O)C2)=O)c(F)c1 C1(C(=O)NCC2CC(NC(c3ncncc3Br)=O)C2)CCC12CCOCC2 C12(NC(c3c(C)noc3)=O)CCCC1CN(C(C1CCO1)=O)C2 C1(N(C(=O)C(C2CC(F)(F)C2)O)C)CCC(CNC(=O)CC2CCC(=O)N2)CC1 c1(NC(c2cc(CNC(C(C3CCOC3)OC)=O)oc2)=O)ccccc1O N(C(=NCC1CCCC1)NCCN1CC(C)CC1=O)C1C(C)(OC(C)C)C1 c1(C(C)=O)cc(C(=O)NCC2(NC(=O)C=C3CC3)CCCCC2C)ccc1O Cc1ccc(CC(N2CC3CC(NC(c4cc(C)c(C)cn4)=O)C3C2)=O)c(Cl)n1 C1(CN(C(CC(C)C2CC2)=O)C2CC2)CCN(C(c2ccccc2C2CC2)=O)CC1 C1(C(=O)OC)CS(=O)(=O)CC1C(=O)Nc1cccc(C(C)(C)C)c1O Cc1cccc(C(=O)NC2CC3C(NC(C4(C)CC5(CCC5)C4)=O)C3C2)c1C Cc1nn(C)c(Cl)c1C(N1CCC(C)(CNC(=O)CCc2cnn(C)c2)CC1)=O C1(NC(c2c(Cl)sc(C)c2C)=O)CCN(C(=O)CC2C=CCCC2)CCC1(F)F c1(C(=O)NC2(C3CN(C(C(CC)C#N)=O)C3)CC2)cc2c(=O)[nH]ccn2n1 c1(CCNC(=O)NC(c2ccccc2)CO)ccccc1Br.C12CC1C2 CCCC(C)CC(=O)N1CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C1 Cc1nc(Br)oc1C(=O)NCC1CCN(C(=O)Cc2cnn(C)c2)CC1 CCC(O)C(F)(F)C(=O)N1CCC(N(C)C(c2nnn3c2CSCC3)=O)C1 c1(NC(=O)N(C2CC3(CNC3)C2)c2ccncc2)cccc(F)c1F c1(C(CC)NC(C2C(C)CN2C(c2nc(C(F)(F)F)cs2)=O)=O)ccc(Br)cc1 c1(OC)cc(Br)cc(CN2CCNCC2C(=O)Nc2ncc(C)cc2O)c1O N1(C(C2CCCN(C(C)C)C2)=O)CC2CCC(NC(C3CC(O)C3)=O)CC2C1 Cc1cc(NCc2cnn(C3CC3)c2)ccc1N(C)C.C1(CC)CCCC1C=O C1(NC(C2CCCN2C(c2nsnc2O)=O)=O)CCn2ccnc2C1 CCCCC(CNC(c1nocc1CC)=O)NC(C1CC=C(C)CC1)=O CC1(C)CN(C(c2cc(C(N)=O)c[nH]2)=O)CC1NC(C1CC2(CC2)CO1)=O CC1CN(C(=O)COCCOCCO)CCC1NC(=O)C(N1CCOCC1)C O(C1CCCc2nccnc21)C(c1[nH]nnc1-c1cccs1)=O CCCN=C(NCCc1ccsc1)NCC1CC1(F)F C1(NC(=O)C=Cc2cocn2)C2CC3CN(C(=O)CC4CSC4)C1C3C2 N1(C(CC2N(C)CCCC2)=O)CC2(CCN(C(c3nc(Br)c[nH]3)=O)CC2)C1 c1(C(C)=O)ccc(NCC(C)CNC(=O)C(O)c2ccsc2)c([N+](=O)[O-])c1 N1(C(C2(CC=C)COC2)=O)CCCC(F)(CNC(c2snc(C)c2N)=O)CC1 N1(C(COCCN(C(=O)C(C)(F)C(C)(C)F)C)=O)CCCC2(CCOC2)C1 C1(C(N2CCN(c3ccccc3)CC2)=O)COCCN1C(C1CC1F)=O c1(CC)ccc(N)c(C(N2CCC(NC(C3CCC4(CC3)CC4)=O)C(O)C2)=O)c1 N1(C(c2c(O)ccc(C(=O)OC)c2)C(=O)NC2CC2)Cc2ccc(F)cc2C1 N1(C(C(CCC)=CCC)=O)CCC(NC(C2CC2c2ccsc2)=O)C2(CCC2)C1 N1(C(C2=CC(C)C2)=O)C2CCC1CC(N(C(=O)C(c1ccc(F)cc1)C)C)C2 CCCCC(C)N=c1nc2scnc2c(NCC2CCN(C)C2)[nH]1 c1(C(=O)NCCN(C)C(C2C(F)(F)C23CC3)=O)ccc(NC(=O)C2CC2)cc1 C1(NC(Cn2c(C)c(Cl)cn2)=O)CN(C(=O)CN2CCNC2=O)CC12CC2 Clc1cc(-c2ccccn2)nc(=NCC2CCc3c[nH]nc3C2)[nH]1 c1(C(C(=O)OC)OC(C2CC(C(=O)N(C)C)C2)=O)cc(Cl)ccc1Cl C1(NC(CCCCC)=O)CCN(C(c2nc(Cl)ccc2F)=O)C12CCC2 c1(C(=O)NCCCOCCN(C(C(CCC#C)O)=O)C)cc2cccnc2[nH]1 N1(C(c2c(C)noc2C(C)C)=O)CCCCC(NC(c2cc(C(N)=O)co2)=O)C1 CC1(C)CCN(CC(N2CCCCC2CCCNC(C2C3CCCC23)=O)=O)C1 C1(CNC(C(=O)NCC)=O)CC(NC(c2sc(C)cc2C)=O)C1(C)C c1(C(=O)NC(CNC(c2cnc(OC)nc2C)=O)(C)CO)nc(C)c(C)[nH]c1=O C123CC(C1)(OC2C)CNC(=O)C=CC(=O)NCC1CN(CC1C)C3=O.CC.CO N1(Cc2cn(C(C)C)nc2)CC(NC(=O)Cc2cc[nH]n2)C(C#N)C1 C#Cc1ccc(C(=O)NC2(C)CN(C(=O)CCc3ccn(C)n3)C2)c(OC)c1 N1(C(C(C)OCC=C)=O)CCOCC1C(=O)NC1CC(N2CCC2)C1 c1(CCN(C2CCN(C(=O)OC(C)(C)C)C2)C(c2ccco2)=O)ccc(F)cn1 N1(C(C2(C)COC2)=O)CCC(CC(=O)NCCC(O)CO)C1(C)C C1(C(C)=O)CC(NC(=O)C=Cc2cnc[nH]2)C1(C)C.N12CC(C1)C2=O c1(C(N(CCCCCNC(C(C2CCC2)OCC)=O)C)=O)cccn2nnnc12 N1(C(=O)OC(C)(C)C)C(C(=O)OCSc2cc(OC(F)(F)F)on2)CC2CCCC12 C1(CCC(=O)N(C(CCCCCCC)C)CCCC#N)Cc2ccccc2CN1 N1(C(c2nc(C)oc2)=O)CCCC2(C1)CN(C(c1csc(CC(F)(F)F)n1)=O)C2 c1(CC(=O)NCCCCN(C(C2CC(CCC)OCC2)=O)C)ccc(C)c(C)c1 CCCCC(CCCC)CC(CC)C(=O)N1CCC(c2cscn2)CC1 Cc1ccc(C)c(C(N2CCCC(C(=O)NC(C)C(N)=O)C2)=O)n1 C1(C(C)C)CN(C(=O)C(N2CCCCCC2)C)CCCN1C(c1cnsn1)=O N1(C(c2c(N)ccc(Cl)c2)=O)CCC2(CCCCC2NC(=O)C(F)CC2CC2)CC1 c1(C(=O)NCCC2(C)CCN(C(c3ccc(OC)s3)=O)C2)ncnc2ccsc12 c1(C(N2C(C(=O)NOCCCCF)CCC(O)C2)=O)c[nH]c2cnccc12 c1(C(=O)NC2C(C(=O)OCC)CCC=CCC2)cc2cc(Br)ccc2o1 CC1(C)CCN(C(=O)CC(Cl)Cl)C1.C1(CC)CCCN(C(C2CCCCC2OC)=O)C1 c1(C(N2CCC(CC=C)(NC(=O)CC(CC)SC)C2)=O)cccc(S(N)(=O)=O)c1C Cn1ncc(CNC(c2cn(CCNC(c3cccc(O)c3)=O)nn2)=O)c1O c1(C(N(CCNC(CNS(CCCC)(=O)=O)=O)CC)=O)nccc2nn[nH]c12 c1(C(=O)NCCOCCN(C)C(C2CCOC2)=O)cc2ccccc2n1C C(=O)(C(C)(C)n1cc(Cl)cn1)NCC(C)NC(=O)CC(c1ccccc1)C1CC1 c1(C(=O)NC(C2CCCC2)CNC(C2C(C)(C)CO2)=O)c(F)ccnc1Cl n1(CCN(C(C2CCc3nnnn3CC2)=O)CC)cnc2c(C)cccc2c1=O c1(C(=O)OC)c(Cl)cccc1S(=O)(=O)NC(C1CCCCO1)C C12(NC(c3cc(C(F)(F)F)ncn3)=O)CCCC1CN(C(c1csc(Cl)c1)=O)C2 C(CN(C)C(c1ncoc1C1CCCO1)=O)(CO)(CO)NC(C(COC)O)=O C1(NC(C2(C)CCCOC2)=O)CN(C(c2cccc(CO)c2)=O)CC2(CCC2)C1 C(=O)(C(C)(C)CCCNC(C1CCC1C)=O)NCc1ccc(OCC)cc1 c1(C(=O)NCC(CC(C)C)NC(C2CC2CN(C)C)=O)ccc(O)c(F)c1F Cc1ccc(C(=O)NC2CC(O)CN(C(=O)C=Cc3cccc(F)c3)C2)c(C)c1 c1(C(N2C(CN(C(C=CCCC)=O)C)COCC2)=O)cc2c(Br)cccc2[nH]1 S(=O)(=O)(c1ccc(C(=O)NCC2CN(C(C3(C(F)F)CCC3)=O)C2)o1)NC CS(=O)(=O)C1CC2CCC(C1)N2C(C1CCc2nc(O)[nH]c2C1)=O C1(NC(c2cccc(C)c2)=O)CCC2(CC1)CN(C(c1cncc(F)c1Cl)=O)C2 C1(C(N(CC(C)(C)NC(c2cccc(CO)n2)=O)C)=O)CCc2ncccc2C1 n1(CC)cc(CC(=O)NC2(COC)CN(C(=O)CCCOC(C)C)C2)cn1 Cc1csc2cc(C(=O)NC(c3cc(F)ccc3F)C(=O)O)[nH]c12 C1(CC)C(C(=O)N(CCOC)C)CCN1C(c1cnsc1)=O Cc1ccccc1CCC(C)CNC(=O)N.C1(C)(N)CCOC1C CCCN(OC)C(=O)CC(C(F)F)NC(c1cc(C)[nH]c1C)=O C(N=c1ccn(CCOC(F)F)[nH]1)(c1cccc(C(C)(C)C)c1)c1cccc(F)c1 C1(C(=O)NCCC2CN(C(c3coc(Cl)n3)=O)CCO2)CC2CCCN2C(=O)N1 C1(C(=O)NC2CCCN(C(C3OCC(C)C3)=O)C2)CC1C1CCCC1 C1(CC(=O)N(C2(CC(=O)NCC(C)CO)CC2)C)CCN(C)CC1 c1(NC(CC)CSC(c2cccc(C(=O)O)c2)C)nc(Br)ccc1C c1(CN(CCCNC(c2cocn2)=O)C(C2CCC3CCC23)=O)ccc(Cl)nc1 c1(C(N2CC(N3CCC3)C2)=O)cccc(C(N)=O)n1.C12CCCC1C(=O)NC2 N1(C(C2(C)CC2)=O)CCOC2(CCN(C(=O)CCNS(=O)(=O)C(F)(F)F)CC2)C1 C(=O)(C1COc2ccc([N+](=O)[O-])cc21)N1CC(NC(CN(C)CCO)=O)C(O)C1 C1(C(N2C(CCC=C)CCC2)=O)(CNC(c2ccnnc2)=O)CC2(CC2)C1 C12(CNC(=O)COCC(c3cccc(F)c3)=O)CN(C(=O)CCF)CC1CCO2 C12(C(=O)NC(c3cn(C)cn3)C)COC(C1)C(NC(C1SCCS1)=O)C2 N1(C(c2cnc(=N)[nH]c2)=O)CCC2CC1CN2C(C1CCCC(F)(F)C1)=O c1ccc2c(c1)C(O)CC1(CC1)O2.c1(CN)nc(Br)ccc1C=O C(C1OCCc2sc(F)cc21)NC(C(n1c(C(F)(F)F)nc2ccccc12)C)=O c1(C(N(CCCNC(C2CC2CF)=O)CC)=O)cc(Cl)c(N)cc1F C1(C(=O)NC(C2CCCC2)CO)CCCCCN1C(=O)Cc1ccsn1 C1(NC(C(C(C)(C)C)O)=O)CC2CCC1CN(C(c1ccc(O)c(N)n1)=O)C2 c1(CCC(N2CC3CN(C(C4CC4(F)F)=O)CC3C2)=O)nc2cnccc2[nH]1 C#CCC(CC(=O)N1CCOC(C(C)N(C)C)C1)NC(C1(CCC)CC1)=O C1(NC(c2cc(Cl)c[nH]2)=O)CC2CC1CN2C(=O)Cc1csc(C2CC2)n1 c1(C(=O)NCC(C(C)(C)C)NC(=O)CC2CCCO2)cc2ccccc2o1 C(=O)(C1(C)CCOc2ccccc21)N1C(CCNC(CCC=C)=O)CSCC1 C(c1c(F)cccc1F)=C(C)C(=O)OC(C)CCc1c[nH]c2ccccc12 c1(C(=O)NC(CCCC)CNC(C2CC2CCC)=O)scc2c1OCCO2 C1(CC)CCCCC1CNCc1ccccc1.C(CC(C)C)N(CC)CC C1(N(C(=O)Cc2csnn2)C)CCC(NC(c2coc(C(F)F)c2)=O)CC1 c1(C(N2C(COC)CC2)=O)cnsc1C(=O)OC(c1nscc1Br)=O CC1(C)CN(C(=O)C2=NNC(C(F)(F)F)C2)CCC1NC(c1cc(O)ncn1)=O c1(CC(N2CC=CC(NC(C(C(C)(C)C)O)=O)C2)=O)cccc2ccncc12 c1(C(=O)NCC2(NC(CC(C)c3cnn(C)c3)=O)CCC2)cnc(C(N)=O)cn1 N1(C(c2c(C)nco2)=O)CC2N(C(=O)C(C)n3ccnn3)CCC2(C)C1 C(CSC)(C(=O)N(C)CCC1CCCCC1)NC(C(C1CCC1)OCC)=O c1(NC(C)C)cccc(C(N2CC=CC2CNC(c2ccn(C)c2)=O)=O)c1 c1(OC)ncc(C(N2CCN(C(C3CC4C=CC3C4)=O)CC2C2CC2)=O)nc1C N1(C(C=C(CC)CC)=O)CCN(C(=O)Cc2nnc(C(F)F)o2)CCC1C CCCCC(O)C(C)C(=O)NCC1CCN(C(=O)CN2CSCC2=O)C1 c1(CN2CC(CNC(c3ccc(Br)cc3O)=O)C(O)CC2)cc(Cl)ccc1F C1(CNC(C2CC(NC(=O)Cc3nccs3)C2)=O)CC2CCC1O2 n1(CCC(=O)NCC2CC(NC(C(C)OC)=O)C2)cnc2c(cnn2C)c1=O CC(C)C(C(=O)N1CC(NC(c2n[nH]c3c2CCCC3)=O)CC12CCC2)C(C)C c1(C(=O)NCC(CNC(=O)C(n2nccc2C)C)OC)cc2ccsc2c(O)n1 Cn1nnc(C(N2CC(NC(=O)CC3CNC(=O)C3)C(O)C2)=O)c1C(F)(F)F C1(CNC(C=CCC)=O)CC(C)(C)CN1C(c1cncc(F)c1)=O N1(C(=O)CC2CCCS2(=O)=O)CCN(C(=O)Cn2nnnc2C2CC2)C(C2CC2)C1 CN1CCCC(CCC(=O)NCCOC2CCN(C(c3cnns3)=O)CC2)C1 C(=O)(CCCCCCOc1cccc2c1COC2=O)OCC c1(C(=O)NC2CCN(C(C(C)OCC#C)=O)CC2)cc(OC)ccc1C N1(C(C(CC=C)(C)C)=O)CCCC(C2CCN(C(=O)CC3CCCC(C)O3)C2)C1 c1(-c2ccnc(NC(=O)NCC3CCC(C)CC3)n2)cc2ccccc2o1 C1(C)(C(C)C)CCN(C(=O)C(C2(O)CCC2)NC(=O)CC23CCCC2C3)CC1 C(=O)(C1Cc2c(Cl)cccc21)NCC1(C)N(C(CCCCCCC#C)=O)CCC1 C(CCOC)(C(=O)NCCCc1ncnn1C)NC(Cc1c(CC)con1)=O C1(NC(c2cccs2)=O)CC2CC1CN2C(c1ccnc(CO)c1)=O N1(CC)N=C(C(=O)NCC=CCNC(=O)CC2CCC23CCOCC3)CCC1=O Cc1c(CCC(=O)NCCC2CCCN(C(c3ns[nH]c3=O)=O)C2)cnn1C O=C(C1=CC2(CCOC2)C1)N1CCC2C(C1)CN2C(=O)C=Cc1cccs1 Cc1ccc2ccc(C(=O)NC3CCC(C(=O)NC4CC4C4CC4)CC3)nc2c1 N1(C(C2C(=C)C2)=O)CC(O)CC1(C)C(N1CCC1C(=O)NC)=O c1(SCC)cc(C(N2CCCC(NC(=O)C(C)(C)CSC)C2)=O)ccn1 c1(C(C)C)nccc(N2CCC(CNC(c3cnn(C)c3)=O)(OC)C2)n1 N1(C(C(COC)COC)=O)CCN(C(=O)CCN(CCC(C)(C)C)C)CC1CO C1(C(=O)NCCOCC)CCN(CCC(=O)NCCc2ccc(C)cc2)CC1O C#CC1(O)CC(C(=O)NC(CCF)C(=O)N2CC(N(C)CCO)C2)C1 c1(C(=O)NC2CC(C)N(C(=O)COC3COC3)CC2)cnc2c(c1)NC(=O)CS2 c1(OCC(=O)N(CCNC(C2(CC)CC2C)=O)C)c(Cl)cc(Cl)cc1Cl C1(n2cc(-c3n[nH]c(C)c3C)nn2)CN(C(C2CS(=O)C2)=O)CCC1O C(=O)(C(C(C)C)n1cnnc1)NCC(C)NC(c1nc(C)[nH]n1)=O C(=O)(C1=NOC(C)(C)C1)N1CCC(C(N2CCC(OCC=C)C2)=O)C12CC2 C(=O)(CCCCCCCO)N1CC2CCN(C(=O)Cc3ccc(Br)cc3)C2C1 C1(NC(C=C(C)C2CC2)=O)CC2CN(C(C3CC(C4CC4)=NO3)=O)CC12 C=CC1(C(=O)NOCCc2ccccc2)CCN(C(c2ncccc2Cl)=O)CC1 N1(C(c2occc2C)C(=O)NCCCCCC)CCC(C2CC(F)(F)C2)C1 N1(C(CC(C=C)(C)C)=O)CCC2CC(C1)CN(C(C1CNC(=O)C1)=O)C2 C1(NC(N(CCCNC(C2(OC(C)C)CCC2)=O)C)=O)CCN(C)C(=O)C1 c1(C(=O)NC2C(CNC(=O)Cc3ccccc3)C2)ccc2c(c1)S(=O)(=O)NC2 N1(C(c2cc(C)n(C)c2)=O)CCC2(CC1)C(NC(c1ccnnc1)=O)CS2(=O)=O C#CCCC(C(=O)NCC1CN2CCC1CC2)NC(c1ncsc1NC)=O c1(C(=O)NCC(CN(C)C(C2(CO)CCCO2)=O)(C)C)cc2n(n1)CCCC2 CCC(CC)C(C(=O)NC1CC2CC1CN(C(=O)COCC(C)C(C)C)C2)OC CC(C)C(F)C(=O)N(C1CCN(C(C2(C(c3ccccc3)=O)CC2)=O)C1)CCO N1(C(c2ccc(CO)cc2Cl)C(=O)Nc2ccccc2)CCc2ccccc2C1 C1(CNC(C(C)=CC2CC2)=O)CN(C(=O)CCC2CC2)C2CC12 C1(NC(c2cnc(C3CCOC3)s2)=O)CCC(F)(CNC(c2ccccc2Cl)=O)C1 N1(C(=O)CCCn2cc(-c3ccncc3)nn2)CCC2(CCCCC2)C(O)C1 c1(OCC(=O)NC(C2CN(C(CCCC)=O)C2)C)ccc(Cl)cc1C c1(C(=O)NC2CCOCC2)ccc(S(=O)(=O)NC2COC23CCC3)cc1 c1(CC(=O)NC2(CN(C(CC3ON=C(C)C3)=O)C)CC2)cnn2c1OCCC2 C=C(C)CCCC(=O)NC1CC(C)(NC(C2CC(C)C2(C)C)=O)C1 C12(C(=O)NCCCCC(C)NC(C(C)O)=O)CC3CC(C)(C1)CC(C)(C3)C2 n1(CCC(=O)NCCC(C)NC(C2CCC3(CC3)C2)=O)ccc(O)nc1=O CCC(COC)C(=O)N1CC2CC1(C(=O)NCC(F)(F)C(C)O)C2 C1(CNC(C(C)Cc2ccnn2C)=O)CC(C2CNC2)C1 C1(CC)CCCCCN1C(C1CCC(CNC(C2CCCN2C)=O)O1)=O C(CC(C)(C)NC(=O)C(C)n1cccn1)N(C(COCCC)=O)C C12(CNC(C3CC(n4cc(-c5cncc(C)c5)nn4)C3)=O)CC1COC21CCC1 CC1CC(NC(=O)CCc2cccc(Cl)c2)CCN1C(=O)CS(=O)(=O)N(C)C C1(NC(=O)Cc2cscn2)CN(C(C2CCCCC(F)(F)C2)=O)C2CCCC12 C(=O)(C(C)C(C)(C)C)N1CCC(O)(CCNC(C(c2c(OC)cccc2)=O)=O)C1 C#CCC(CC(F)F)C(=O)N1CC2CCCCC2(NC(=O)C(COC)CC)C1 c1(SCC)cccnc1C(=O)NC1CC(C(=O)NCCCCCF)C1 N1(C(c2scc(NC(C)=O)c2)=O)C2CCC1CN(C(=O)CCNC(=O)CO)CC2 N1(C(=O)OC(C)(C)C)CCCC(OC2CC(NC(C3CCOCO3)=O)C2)C1(C)C C1(F)(C(=O)NC2CCC(N(C(c3cnc(C)nc3C)=O)C)C2)CCC(F)(F)CC1 C12(COC)CN(C(=O)Cc3cnn(C)c3)C(CNC(C3(C)CC(F)(F)C3)=O)(C1)C2 c1(C(N2CCC(C(CNC(CCC#C)=O)F)CC2)=O)cc(F)c(F)cc1N C1(C(N(CC(CCC)C)C)=O)CC2CC1CN(C(C1CC1C(C)C)=O)C2 C1(C)(C(=O)NCC(=C)CCNC(c2ccns2)=O)CCOC(C)C1 c1(C(N2CC(NC(C34CCN(CC3)C4)=O)C(O)C2)=O)ccc(F)c(F)c1F N1(C(CSCC#C)=O)CCCC(NC(c2cc(SC)c(C)o2)=O)C1C N1(C(CCc2nc(C)sc2)=O)CC2CCC1C1CN(C(c3ccon3)=O)CC21 N1(C(c2c(C)c(Cl)ccn2)=O)CCC(NC(C2CCCS(=O)(=O)C2)=O)C12CCC2 CC1(C)C(CC(=O)NCCC2CCN(C(c3cccnc3S)=O)CC2)CC1O C(C(=O)NC(c1ccccc1)CNC(=O)C(CCO)N(C)C)(C(C)C)OCC N1(C(C2C(C)CCC2)=O)CC=C(CCNC(c2ccc(C(C)(C)C)[nH]2)=O)CC1 c1(CC)nc2sc(C)cn2c1C(=O)NC1CN(C(=O)Cn2cccn2)CC1C N1(C(=O)OC(C)(C)C)CCCC(C)(CNCc2ncc(Cl)s2)C1 c1(C(N(CC(C)NC(C(c2ccccc2)C)=O)C)=O)c(F)ccnc1Cl c1(C(N2CCN(C(c3c(C)nco3)=O)CC2C(C)C)=O)ccn2c(C)cnc2c1 CCC(CC(=O)N1CC(C)CCC1CNC(=O)C=Cc1cn(C)nn1)C(C)(C)C C1(C(N2C(C)CN(C(c3ccc(O)nc3)=O)CC2)=O)CC(C2CCCC2)C1 C(C(C)(O)CC(=O)N1CC(C(C)NC(=O)CCCNc2ccccc2)C1)OC C(=O)(CC(C)P(C)(C)=O)NCCOCC(N1CC(O)(CC=C)C1)=O c1(NC(C(C(C)C)C)CNC(C2(Br)CC2)=O)ncc2ccsc2n1 c1(C(=O)NC(C2(O)CN(C(c3c[nH]ccc3=N)=O)C2)C)cc2nnn(C)c2s1 C1(CNC(C(CC)F)=O)CC2(CCN(C(=O)CC3CCCC(=O)N3)C2)CO1 C1(N(C)C(C2CC=CCC2)=O)CC2CC1N(C(=O)Cc1cncs1)C2 c1(CC)ccc(F)c(C(=O)NC2COCC2NC(=O)C(=O)NCCSC2CC2)c1 C1(NC(C(CCC)NC(=O)CCc2ncnn2C)=O)Cc2cscc2C1 c1(C(=O)NC(C)(C)CNC(C2(CO)CCC2)=O)nc(Br)c2ccccn12 c1(CC(=O)N(C)CC2(NC(C(c3cccs3)SC)=O)CC2)conc1C C(=O)(C(C(C)C)c1ccn(C)n1)N(CCNC(c1ccc(C(=O)OC)o1)=O)CC CCC(C)C(CC(=O)NC1(C2CCCO2)CC1)NC(=O)CS(C)(=O)=O Cc1c(C(N2CC3(CC(NC(=O)CNS(N)(=O)=O)C3)C2)=O)cccc1Cl c1(C(=O)OC)ccc(C(N2CCC(CC3CCC(C)C3)C2)C(=O)NC(C)C)o1 C1(CNC(c2n(CC)cc(Cl)c2)=O)C(C2CC2)CCN1C(c1cnnc(Cl)c1)=O N1(C(=O)OC)CC2C=CC1C(C(=O)NC1CC(O)(CC(C3CCN3CC)=O)C1)C2 CCCCC(=O)NC1(C2CCCN2C(c2cc(C3CC3C)on2)=O)CC1 C(=O)(C(C)C(O)CCCC)NC(c1cn(-c2ccc(C)c(C#N)c2)nn1)CCC C(=O)(CC(C)(F)F)NC1CC(OCC(=O)NC(C2CCCCO2)C)C1 N1(C(CC=CCC)=O)CCC(CO)(NC(c2nc(C(F)(F)F)cn2C)=O)CC1 CC1(NC(c2coc(Br)n2)=O)CCCN(C(C2(C3CCCO3)CCC2)=O)C1 C1(C)(NC(c2c(C)n(C(C)(C)C)nc2)=O)CCCN(C(=O)NC(C)(C)C)C1 c1(C(N2CC(C)(C)C(NC(=O)CCS(N)(=O)=O)C2)=O)ccc2c(c1)COC2 c1(COC)ccnc(C(N2CC3CC2C3NC(C2CCOC2C2CC2)=O)=O)c1 Cc1cc(C(=O)N(CCN(C)C(c2snnc2C2CC2)=O)C(C)C)nn1C(C)C c12cc(cc(Cl)c1)CC(=O)N2.N1(C(C(C)S)=O)CCCC(Cn2ccnc2)C1 CCCCC(CNC(=O)CCCC1CCCO1)NC(C1CSCC(=O)N1)=O C1(CNC(C2(N(C(c3n(C(CC)C)ncc3)=O)C)CC2)=O)CCCCCC1 c1(C(=O)NC(C(CO)NC(CCc2c(C)n[nH]c2C)=O)C)coc(S(N)(=O)=O)c1 N1(C(C2(COC)CCCO2)=O)CC2=C(C1)CN(C(C1(F)CCS(=O)(=O)C1)=O)C2 N1(C(C=Cc2occ(C)n2)=O)CCOC2CN(C(C3CC3(F)F)=O)CC12 c1(C(N2CCC(CN(C)C(C3(O)CCSC3)=O)C2)=O)cc2cc(F)ccc2[nH]1 CC(=O)CCCC(=O)NCC1CCN(C(C2C3(CC3)C23CC3)=O)C12CC2 CCC(C#N)(CC)C(=O)NC1COCCN(c2cc(C(N)=O)ccc2[N+](=O)[O-])C1 C(=O)(CCCC(=O)N1CCC(C(C)C(=O)N(C)Cc2ccc(Br)cc2)C1)OC N1(C(=O)NC2(COCC)CCCC2)CC(C(C(=O)Cc2c[nH]nc2O)=O)C(C)C1 C(C1=CCN(C(=O)CC2CCC(F)(F)CO2)CC1)NC(c1c(C)nns1)=O Cc1cc2cc(C(=O)NC3C4CCC3N(C(C3CCSC3)=O)C4)c(Cl)cc2[nH]1 Cc1ccc(CC(=O)N(CCNC(C2C=CCC2)=O)CC2CC2)cc1 CC1CCCN(C(=O)CN(c2cnn(C)c2)C)C1CCNC(=O)C(=O)N(C)C C(CCCC(CO)NC(c1cc(C2CC2)ccn1)=O)NC(CC(=C)C)=O S(=O)(=O)(c1cccc(NC2CCCN2S(C)(=O)=O)c1C)NC Cc1cnc(C(=O)N(C(C)CN(C)C(c2nc(C(C)(C)C)no2)=O)C)c(C)c1 S(=O)(=O)(c1nccs1)N1C(C(=O)NC2CS(=O)(=O)C2)CCCC1 N1(C(c2c(OC)n[nH]c2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)C(C2CC2)C1 CCN=c1[nH]c(C(=O)NC(CCN(C(=O)Cc2cccnc2O)C)C(C)C)cs1 c1(C(CCO)NC(=O)Nc2ccccc2-n2cnnn2)ccc(Cl)c(F)c1 c1(C(=O)NC(C)C=CC(=O)NC(c2ccncn2)C)ncncc1Cl c1(OCC(=O)NCC(O)CCc2ccccc2)ccccc1Br c1(C2(CCC(=O)NCCCN(C(C=C(CC)C)=O)C)CC2)ccccc1 c1(C(=O)OCC)ccc(C(=O)NCCCC(C)NC(=O)Cn2cc(C)cn2)cc1 C1(NC(C2N(C(C(CC(N)=O)O)=O)CCCCC2)=O)CCC2(CCCC2)C1 C1(C#N)(C(N(C)CC2N(C(COCCCC#C)=O)CCCC2)=O)CCCOC1 N1(C(C(=O)NC2CCC(C(C)C)CC2)=O)CCCC(CN)C1C C(=O)(C1=NOC(C)(C)C1)NCCCCN(C(c1ccc(C)c(Br)c1)=O)C c1(C(=O)NC2CC(C(=O)NC(COC)C3CC3)OCC2)cnc(C)c(C#N)c1 c1(NC(N2C(C(=O)NC34CC(C(=O)OC)C3C4)CCC2)=O)ncccc1Cl C(=O)(CS(=O)(=O)CC(=O)NCC1COCC1NC(c1cc(C)n(C)n1)=O)OC c1(C2(C(=O)NCCCNC(C(C)C3CCCC3)=O)CC2)cccc(F)c1 C1(C2CCCN(C(=O)C(C)(C)C(F)F)C2)(NC(c2c(C)[nH]nc2C(F)F)=O)CC1 C1(C(N2C(CNC(C(F)=CC)=O)CC3(CCC3)C2)=O)Cc2cccc(C)c2O1 c1(C(=O)NCC(CCOC)NC(C2CCC(C)O2)=O)cc([N+](=O)[O-])cn1C C12(CNC(CC3CN(C)C3)=O)CCC(C1)N(C(=O)CCn1cc(Cl)cn1)C2 C1(C(=O)NCCCC(=O)OCC)C2CN(C(=O)N(C)C3CC3)CC12 Cc1cc(CN2CCC(O)(C(=O)NCc3ccc(Br)cn3)C2)ccc1[N+](=O)[O-] c1(CNC(CSCC=C)=O)ccccc1NC(=O)C(=O)NCCOC N1(CC)CC(O)CC1(C)CNC(=S)NC1CCNC2(CC2)C1 CC(C)C(O)C(=O)NC(C(=O)NCCOCCCO)c1ccco1 c1(OCCCC(=O)NCCn2ncc3ccccc23)nc(Cl)c(Br)cc1I c1(Cc2n(CC(C)C)c(N3CC4(C)COC4C3)nn2)noc2c1CCCC2 c1(CCC)c(C(=O)NC2(C)CC(NC(C3CCCCC3OC)=O)C2)nnn1C CCC(C)CCC(=O)NCC1CCC1NC(c1coc(C(C)C)n1)=O C(C(F)F)(C(C)(C)C)NC(CC(C1CC1)NC(C1C(C)CCO1)=O)=O N1(C(C(=O)NC(C)C)=O)CC2(C1)CN(C(c1occc1Cl)=O)CCO2 Cc1ccc(CC(N2CCC(O)(CN(C(=O)C(F)(F)CC3CC3)C)C2)=O)cc1C C1(C)(C(N2CC(N(C(CNC(C3C(C)C3)=O)=O)C)C2)=O)CCNC1=O C(=O)(CCS(C)(=O)=O)NCc1cccc(C(=O)N(C(c2noc(C)n2)CC)CC)c1 N1(C(C)C)CC(C(=O)NCCC2CC(NC(=O)Cc3ccc(F)cn3)C2)CC1=O C=C1CCN(C(=O)C(C2CC2)C2CC2)C(C(=O)N(C)Cc2ccccc2C)C1 C1(C)(C(=O)NCCNC(C)=O)CC1(F)F.C1(=O)C(=O)NC(CO)CN1 c1(C(N2CCN(C(C3N=C(C)SC3)=O)C(C)C2)=O)noc2c1CCCCC2 C1(NC(C(C2CCOC2)OCC)=O)(CC)CCN(C(c2cnc(CC)o2)=O)CC1 c1(C2CCN(C(=O)OC(C)(C)C)CC2)nnc2n1CCN(C(C1CC(=O)N1)=O)C2 CCCS(=O)(=O)C(C)C(=O)NCC1CCCC1NC(=O)Cc1ccc(C)nc1 O=C(N=c1c(Cl)c[nH]cc1Br)c1n[nH]cc1NCC1CCC(F)(F)CC1 CCC(C(=O)N1CCC(C(C)NC(=O)CC2(O)CCOC2)C1)C(C)C c1(CC(=O)N(C(C)CNC(CCCc2onc(CC)n2)=O)CC)cccc(C)c1 CC1(C)COC(CCC(=O)NCCC2CC(NC(c3cnn(C4CC4)c3)=O)C2)C1 C(=O)(C(C)C(C)NC(c1ccc(=O)oc1)=O)NC(CC(=O)OCC)c1ccccc1 c1(C(=O)NC(COC)C)csc2c1CCN(C(=O)C(=O)c1ccco1)C2 C=CCCCCC(=O)NCC(C)(C1CC1)NC(C1CC(OCC2CC=CCC2)C1)=O N1(C(C(n2cc(C(=O)N(C)CCF)nn2)C)=O)Cc2ccccc2C1 N1(CCNC(C)C#N)CCC12CCCC(C)(C)C2 FC1(F)CCC(CSCCNC2CCCNC2)C1 N1(C(C(CSC)O)=O)CC2(C1)CN(C(=O)CC1=CCCC1)CCO2 c1(COCC(=O)NCC(C)(C2CCC2)NC(C2C(=C)C2)=O)cccnc1 C12(CCCCC1)C(=O)N2.CC1=NOC(C(=O)NN2CCC(n3cccn3)C2)C1 N1(C(=O)C=Cc2ccccc2[N+](=O)[O-])CCN(C(=O)CCCC(N)=O)CC(O)C1 c1(C(=O)NCC2(CNC(C3C(CC)C3)=O)CCCC2)cccc(C2CC2)c1N c1(OC)cnc(F)c(C(N2CCCCC2CNC(c2c[nH]c(=N)nc2O)=O)=O)c1 C1(C(=O)NCCCc2scc(C)n2)CCCN(C(c2ccn(C)n2)=O)C1C N1(C(CCC(CC)C)=O)CCC2CN(C(c3cn4ccnc4s3)=O)CC2C1 CCC(CC)C(=O)NC(C)CCNC(c1ccc(I)cc1)=O C(=O)(C(C)CC(C)C)N(CC(=O)N(CC=C)CCOC)C C(=O)(C1CCCc2nccn21)N(C(C)CCNC(=O)CCc1ccc(F)cc1)C C1(NC(C2C(=C)C2)=O)CCN(C(=O)C=Cc2ncc[nH]2)CC1O CCCC(C)CCCC(=O)N1CCC(CN(C(=O)C2=COCC2)C)C1 CC1CCN(C(c2ccnc(C(C)C)n2)=O)CC1NC(=O)C(C1CCOCC1)F Brc1ccc2c(N3CCCC3Nc3ncnc(N4CCCC4)n3)ncnc2c1 C(CNC(=O)C1=CC(C)(C)C1)(C(C)C(C)C)NC(CCC(=C)Br)=O C1(NC(COC)=O)CCN(C(=O)CCc2csc(C)n2)C12CC2 N1(Cc2c(OC)cco2)C2CCC1CC(c1ncco1)C2.C12CCCC1C(=O)N2 c1(C(=O)NC(C)(CNC(=O)CCSc2ccccn2)C2CC2)ccc(C#N)cn1 N1(C(c2cc(C)c(Cl)nc2)=O)CCC2(C1)CN(C(c1ccn(C)n1)=O)C2 Cc1cc(N(C)Cc2ccc(Br)o2)nc(NC2CCCC(CC(N)=O)C2)n1 c1(OC)ccc(-c2cncc(C(=O)Nc3ccc(CO)nc3)c2)c(OC)c1 c1(C(N2C(CN(C)C(C3CC3c3ccco3)=O)CCC2)=O)ccccc1C(F)F c1(CC(=O)NCC#CCNC(CSCC(=O)OC)=O)ccc(Cl)cc1Cl C(=O)(C(O)CCc1ccccc1)N1CC(C(C)NC(=O)CCN2CCC2)C1 C1(CNC(C2CCC3(C2)CC3(F)F)=O)CC2(CCN(C(=O)CC3CC3)CC2)CO1 C1(C(C)(C)C(=O)NCC=CC2CC2)CCN(C(=O)CCC2CCC(=O)C2)CC1 C1(C(=O)NC2CCN(C(CC=CC)=O)C2)CC12CCSCC2 c1(C(=O)NC2C(NC(c3cc(C4CCC4)on3)=O)C2)cccc2ccc(O)nc12 C(=O)(C(C)(C)C(N)=O)NCC1C(NC(CC(CC)C)=O)CCC1 C(=O)(C(F)(F)C1=CCOCC1)N1CCCC(NC(C2(OC(C)=O)CC2)=O)C1 Cc1cccc(C(=O)NC2CCC(N(C)C(c3ccnc(O)c3)=O)C2)c1N C1(CCNC(COCC#C)=O)CN(C(=O)CCC(=O)c2cccnc2)CCO1 C1(C(N(CC(C)(C)CNC(c2cnccc2C#N)=O)C)=O)CCN2CCCC2C1 C1(C(=O)Nc2ncccc2CO)CC(F)CN(C(c2cncc(F)c2)=O)C1 N1(C(CCN(CC=C)C(c2cnc(O)c(F)c2)=O)=O)CCC(CO)C(O)C1 c1(N2CCC(CCNC(=O)C(F)C(F)(F)F)C2)ncc2ccnc-2[nH]1 c1(-n2ncc(C(N3CC(NC4CC4)C3)=O)c2C(F)(F)F)cc(Cl)ccc1Cl N1(C(c2ccc(CCC)s2)=O)CCC2(NC(C3(C)CCCOC3)=O)CCCC12 N(C(=NCC(F)(F)c1ccc(C)cc1)NCC1CCOC1)C(C)CC(F)F CCCCCCCC(F)C(=O)NC(CN(C(C1C(C)(C)C1(F)F)=O)CC)CC c1(OCCC(=O)OCC2CCC(=O)N2)cccc([N+](=O)[O-])c1 CCCCCC(=O)NC1CCCN(C(=O)CC2(C(F)(F)F)CNC(=O)C2)C1 O=C(CCCCNC(C1C=CC(COC2CC2)C1)=O)NOCC(F)(F)F C(=O)(CC(C)(C)C(F)F)NC(C)CCCCNC(=O)Cn1cccn1 C1(CCOC)(NC(=O)C(C)OC)CCN(C(C2CC(OC)C2)=O)C1 C(=O)(C(C)CC(N)=O)NCCCCC(C)NC(c1ccc(-c2ccco2)o1)=O N1(C(COCCC#C)=O)CCC2C(CCCN2C(=O)CC2CSC2)C1 N1(C(C2CCN(C(Cn3nc(C)c(Cl)c3)=O)CC2O)=O)CCc2cnccc2C1 N1(C(C=C(C)CNC(c2cc(CO)on2)=O)=O)CC(CO)C1(C)C C(=O)(C#CC1(CSC)CC1)NCC(CCCCSCCC)O.c12ccc(o1)C2 N1(C(Cc2cc(C)cc(F)c2)=O)CCC(F)(F)C(CNC(C23COCC2C3)=O)C1 CC1(C(N2CCN(C(c3ccns3)=O)C(C3CCCC3)C2)=O)CC2CCC1O2 Cc1cccc(OCC(=O)NC(C)(CNC(=O)CC23CC(C2)C3)CO)c1 c1(C(N2CCC(C3CCCCC3)C2)C(=O)NCCC)cc(Br)cc2nc[nH]c12 C(C(O)CC(=O)N(C)CC1CCOC1C)NC(C(C)OCCCC)=O CC(C)CC(C)(CNC(c1ccoc1Cl)=O)NC(=O)C(C)CC1CC1 c1(C(=O)NC(C(=O)NC2C(CC)CCCC2)CCOC)cnccc1C#N CCC(O)C(C)C(=O)NCC1CN(C(=O)CC2CCCC3CC23)CCCO1 N1(C(c2cnn(CC(F)F)c2)C(=O)NCCOC)CCC(C)(O)C1 N1(C(c2c(Cl)nc(OC)s2)=O)CC2ON=C(CNC(=O)C(=O)N(C)C)C2C1 C(=O)(C(C)(C)CC(=O)NC1CCCCC1CNC(c1cnn(CCO)c1)=O)OC c1(C(=O)NC(CCNC(CCC(=C)C)=O)C)cc(OC)ccc1F C(C(C)(C)CN)N(C(c1ccc(F)o1)=O)C(c1cc(-c2ccco2)c[nH]1)=O.CO c1(OC(C)C)ccc(C(N2CC(CNC(=O)CN(C)C)CC2(C)C)=O)c(Cl)c1 c1(C(N2CCC(CCNC(C(C)CC3CCC3)=O)C2)=O)cc2cccc(Cl)c2o1 N1(C(c2ncn(CC)c2)=O)CC(F)(F)CC1C(N1CCOC(C)CC1)=O C1(NC(C(=O)NCC(F)F)=O)CN(C(=O)Cn2cnnc2O)C2CC12 c1(C(=O)OC)cc(C)cnc1N1CC2CC(NC(C3C(C)OC(C)C3C)=O)C2C1 c1(C2CCCN(C(=O)NC(c3ccc(Cl)cc3)C#C)C2)cccc(C#N)c1 C(=O)(C(C(=O)OCC)C(C)C)NC12C(CN(C(CC=CCC)=O)C1)C2.OCC Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)NC(=O)C(CN)C(C)(C)C C1(CNC(C2CCCN(C(c3c(OC)cccc3)=O)C2)=O)CCC2(CCC2)N1 CC1CC(c2nnnn2C2CCC2)(NCC2C(C)(C)C2(C)C)CS1 C(=O)(C1CCCc2cc(C#N)ccc21)N1CC(NC(=O)CCCF)CC(C)(C)C1 C1(NC(CCSCC(N)=O)=O)CC(NC(C2CC3(CC3)C2)=O)C12CCC2 CC(C)CCC(F)C(=O)NC1CC(O)C1CC(=O)NC12CCN(CC1)C2 c1(NC2CC(NC(Cc3n(C)ccn3)=O)C23CCC3)ncc(S(C)(=O)=O)cc1Cl c1(C(=O)NCCCOCCCNC(c2nc(=N)[nH]cc2)=O)ccc(CO)cc1F CN=c1nc(C(N2CCCC(N(C)C(c3cncn3C)=O)CC2)=O)cc(C)[nH]1 C1(C(C)C)CNC(=O)CN1C(=O)Nc1nccn1Cc1ccc(Br)s1 c1(-c2c(OC)cc(C(N3CC4CC4C3C#N)=O)cn2)cnc2n[nH]cc2c1 C(=O)(C(C)C(O)C(C)C)NC1CCN(Cc2cn(-c3ccc(C)nc3)nn2)C1 CCC(C(=O)NC1CCCC1NC(C1(C2CC2)CC=CC1)=O)C(F)(F)F N1(C(C2(C)CCOCC2)=O)CC2CC(NC(=O)CC3CCCCC3(C)C)CC1C2 N1(C(CC2(OC)CCCC2)=O)CCCC(N(C(=O)Cc2nc(C)c(C)[nH]2)C)C1 C(=O)(CC(C)P(C)(C)=O)N1CC(C(C)C)N(C(C2CCCC(=O)CC2)=O)CC1 C(CCCCCCCO)NC(C1N(C(c2c(C)ccc(O)c2)=O)CC(F)(F)C1)=O C12(NC(c3ccc(CC)s3)=O)CCC(C1)N(C(=O)Cn1cc(C3CC3)nn1)C2 S(=O)(=O)(c1cc(F)cc(F)c1)NC1COCCN(C(c2c(OC)csc2)=O)C1 Cc1ccc(CC(N2CCC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C(F)C2)=O)cc1F c1(C(=O)NC(CC)(C)CNC(c2cc(Cl)ncc2O)=O)cc(C)cc2c1OCC2 N1(C(c2ccn(CC)c(=O)c2)=O)CCC2CN(C(c3cc(Cl)ns3)=O)CC12 O=C(NOCC(N1CC(F)C(F)C1)=O)C1=CC2C=CC1C2 c1(COCC(=O)NC2CCN(C(C)C)CC2)cc(O)cc2ccccc12 CC(CN=c1nc(O)c2c(ncn2C)[nH]1)N(C(=O)CC1CSCCS1)C CCCCCCC(=O)N1CC2CC1C2NC(c1ccoc1Br)=O CC(C)C(C(=O)NCC1(NC(=O)CCc2ccccc2Cl)CCOC1)C1CCC1 c1(C(NOCC(CC)C)=O)cn(CCNC(=O)CCC2CC(OC)C2)cn1 C(=O)(CS(=O)(=O)C1CC1)N1CCCC(C)(NC(C2(C3CCCO3)CC2)=O)C1 N1(C(c2cccc(C)c2C)=O)CCCN(C(c2nocc2Br)=O)C(C)C1 CC(C)CC(C(=O)N(C(C)CNC(C1CC(=O)CC(=O)C1)=O)C)C(N)=O C1(NC(C2N(C(c3cccc(F)c3O)=O)CCC(C)C2)=O)CCCC(C2CC2)C1 CC1(C)CCC2(CC1)CC2C(=O)NCC1CCN1C(=O)CC1CC=CCC1 CCCC(C#N)C(=O)N1CCOCC(NC(c2ccc(CNC(C)=O)o2)=O)C1 c1(C(N2CCC(c3ccccc3)(C(=O)OC)C2)=O)cc(Cl)cnc1F c1(SCCC(=O)NCC(C)NC(=O)CC2CCN(C)C2=O)ccc2c(c1)OCO2 C1(CNC(=O)CCCCCF)CC2COCC2N1C(c1ccc2sncc2c1)=O C1(C(N(C)Cc2ccc(C)cn2)=O)CC(O)CCN1C(=O)CCc1ccn(C)n1 C1(CNC(C(CO)NC(C(C)C)=O)=O)N(C(=O)C(=Cc2cscn2)F)CCC1(C)C c1(OC)ccc(CNC(=NC)NCC2CCCC(C)C2)c(O)c1 N1(C(c2cnc(NC(C)=O)o2)=O)CC=CC(NC(c2nsnc2O)=O)C1 C(=O)(C1=CCCOCC1)N1C(C=CC(=O)NC2C=CC(C(=O)NC)C2)CCC1 c1(-c2cn3cnc(C(N(CC)Cc4ccccn4)=O)c3s2)cccc2c1CCC2 CN1C(=O)CCCC1C(N1CCC(NC(c2cc(C3CC3)no2)=O)C1C1CC1)=O N(C(=NCCCF)NCc1ccnc(OC2CC2)c1)Cc1cc(C(C)(C)C)on1 C1(NC(C=CC(CC)=CC)=O)CCCN(C(=O)CC(C)(C)C2CC2)CC1F C1(C(=O)NC(C)CCF)COC(CNC(C2SCCS2)=O)C1 N1(C(C=CC)=O)CCCC(CN2CCN(C(c3c[nH]c(=O)cn3)=O)CC2)C1 CC1(C)CCC(C(=O)NCC(C)(O)C(F)(F)F)CN1C(=O)CCP(C)(C)=O c1(C2(C(N(CCNC(C3=C(C)CCC3)=O)C)=O)CC2)ccc2c(c1)OCCO2 c1(C(N)=O)ccc(CC2CC2)c(C(F)(F)F)c1.c12ocnc1CC(=O)N2 CCCCC#CC(C)(C)NC(C1CC(NC(=O)C(CC)NC(C)=O)C1)=O Cc1ccc(F)c(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)O)c1 C1(CNC(COCCCC)=O)CCN(C(c2ccsc2Cl)=O)CC1O C(C1=NOC2CN(C(c3nccnc3N)=O)CC12)NC(CC(C(C)C)C(C)C)=O Cn1cnc2nc(N3CCC4(CC3)COC4)nc(N3CCN(CCO)C(C)(C)C3)c12 C1(NC(CP(C)(C)=O)=O)CC1C1CCN(C(C2CCCCC(=O)N2)=O)CC1 c1(C(N2CC(OC)C(F)C2)C(=O)NCC2CC2)ccc(F)c(C(F)(F)F)c1 CCC(C)CC(C(=O)NC1COCC1CN(C)C)NC(c1ccc(F)nc1)=O C1(C(=O)NC2CCCNC2)Cc2ccc(F)cc2C1 c1(C(=O)NC23C(CN(C(C(C(=O)OCC)(C)F)=O)C2)C3)ccc([N+](=O)[O-])cc1F N1(C(CCC(C)(C)O)=O)CCC(C2CCN(C(c3ccncc3)=O)CC2)CC1 C(C(O)C(C)(C)O)OCCNC(CCN(C(C1C(CC)OCC1)=O)C)=O c1(C(=O)NC2CN(C(C(C)=CC)=O)C(C)CC2)[nH]c2ccc(OC)cc2c1C C(=O)(CCCC(F)(F)Br)NC1C(C(=O)Nc2ccc(CO)cn2)CCC1 N#Cc1cccc(CC(=O)OC2CCCN(C(C3(C(=O)N(C)C)CC3)=O)C2=O)c1 C1(NC(c2cnn(CC)c2Cl)=O)CN(C(=O)C(N2CCNC2=O)C)CCC1CO C12(CNC(C3CCC(O)C3)=O)CCC(CC1)N(C(C1(c3ccno3)CC1)=O)C2 c1(C(N(NC(=O)NC(C(=O)OC)C(C)OC(C)=O)C)=O)cc(=O)cc(Cl)[nH]1 C(C(=O)N=c1cc[nH]cc1Cl)C1CCC(NC(C(C)Oc2ccccn2)=O)CC1 c1(C(=O)NCC(C)C(=O)NC2(C)CC2(C)C)ncncc1N Cc1ccc2c(C(=O)NC(CNC(C3CCO3)=O)C(C)(C)C)c[nH]c2c1 c1(CC2(C(N3CCC(NC(=O)C=Cc4cn[nH]c4)C3)=O)CC2)ccc(Cl)cc1F c1(CN2C(C(N(CCCCCO)CC)=O)COCC2)cc(Br)ccc1[N+](=O)[O-] C1(CN(C(=O)Cc2cccc(F)c2)C)CCN(C(C2(C#N)CCOC2)=O)CC1 C(=O)(CC(C(=O)N1CCN(C(c2nnn(C(C)(C)C)n2)=O)C(CF)C1)OC)OC Cc1sc(NC(=O)C(CCN(C)C)NC(C)C(C)C)c(C)c1C N1(Cc2c(SC)c(F)ccc2F)CCC2(CCCN2C(=O)C(C)=O)CC1 CC(C(=O)NCCCCC(=O)NC1CCCC(F)(F)C1)C(F)(F)F CC1(C)CC1(C#N)C(N1CCC(CCC(=O)NCC2(F)CC(O)C2)C1)=O C1(O)(CNC(C2CC(C)(C)C2)=O)CCCN(C(=O)CCOC2CCOC2)CC1 Cn1ncc2c1CC(CCC(=O)OCC(c1cccs1)=O)CC2 C(=O)(CCCC(=O)Nc1nccs1)NC1CC(CNC(c2cc(OC)ns2)=O)C1 CC1CC2(CCN(C(=O)Cn3ncnn3)CC2)CN1C(=O)CCCCCN(C)C Cc1ccc(CNC(=O)CC23CCCC2C3)cc1 C(=O)(C(F)(F)CC(=O)OC)N1C(C)CCC(Nc2ncc(C(=O)OCC)nc2)C1 c1(C(N2CCC3(NC(C=Cc4n(C)ncc4)=O)C(C2)C3)=O)cc(S(N)(=O)=O)co1 C=CCC(C(=O)NC(CNC(C1CC1C(C)C)=O)C(C)C)NC(=O)OC(C)(C)C Cc1sc2ncnc(N3CCC4CCC(C3)N4C(=O)CCOC(C)C)c2c1C N1(C(C=CCOC)=O)CC2CCOCC2(NC(=O)CCc2nncs2)C1 N1(C(CN(CC)CC)=O)CCN(C(c2ccc(C(C)=O)cn2)=O)C2CCCC12 Cc1cnn(C)c1CN(C1COC(C(=O)O)C1)C(C1CC1)C1CC1 C#Cc1ccc(F)c(C(=O)NC2CCCN(C(=O)CC(CC)C(C)C)CC2)c1 N1(C(c2cc(CC)c(F)cc2)=O)CC2OCCN(C(=O)CSC3CC3)C2C1 c1(CCC(=O)NCC(CC)NC(=O)C(O)C2CC2)ccc(OC)cc1OC C1(C(N(CCC(=O)NCC2CCC(CO)CC2)C2CC2)=O)CC2(CCCO2)C1 C1(CCN(C(C2C(C)CC2)=O)C)CCN(C(c2csc(-c3cccs3)n2)=O)CC1 C(=O)(C(F)(F)C(C)O)NCC(C)CC(=O)Nc1cccnc1 N1(C(C2CCS2(=O)=O)=O)CC2CCC1C(N=c1c(Cl)c[nH]cc1[N+](=O)[O-])C2 C1(C(N(CCCCNC(=O)CCCc2csc(=N)[nH]2)C)=O)CC2CCCCC12 C(=O)(CCC(=O)NC(C1CC(NC(C2(C(=O)NC)CC2)=O)C1)C)OCC C12(OC)CCC(C(=O)NC3CCN(C(C4CCC(=O)O4)=O)CC3CO)(CC1)C2 C1(C(=O)NC2C(CNC(C(CC)(C)C)=O)CCCC2)CC2(CCC2O)C1 n1(C(C(=O)OC)C)nnnc1C(COc1ccccc1)NCc1coc(C)n1 C1(C(=O)NCC(C)NC(C(C)(C)NC(=O)NCC=C)=O)CCCOC1C c1(OC)ccc2[nH]c(=NCC3CSCCS3)[nH]c(=NCc3conc3Br)c2c1 c1(C(N2CC(CCNC(=O)NC(C)C(=O)NC3CC3)C2)=O)cc(C(F)(F)F)cs1 N1(C(CN(C(=O)NCC2CC2c2ccccc2)C2CC2)=O)C2CCCC1CC(O)C2 C12(CNC(c3cccc(=O)o3)=O)CN(C(c3ccnc(S)c3)=O)CC1CCO2 C1(CC)(CO)CN(C(=O)C(C2(O)CCC2)NC(C2CCC(=O)N2)=O)C1 C12(O)CC(C1)CNC(=O)N(C1CCOC1)C2.C(C)(C)(C)OCCOC C(C(C)C)(C(O)C(=O)N(CCNC(c1ccn(CC(C)C)n1)=O)C1CC1)OC C1(C)(OC(C)C)CCN(C(=O)CCNC(=O)C(C)C(F)F)CC1 c1(CCN=C(NC2C3(CC(OCC)C3)C2)NC2CC2)ccc2ncccc2c1 c1(C(N2CCC(NC(CCCn3ncc(C)c3)=O)C2C)=O)cncc(N(C)C)c1C c1(C(=O)NC2C(NC(c3nc(CC)oc3C)=O)COC2)ccc2nc(O)sc2c1 Cc1c(CC(=O)N(CCCN(CCCNC(=O)CC2CCC2)C)CCO)cnn1C CCC(C)CCCC(=O)N1CC(NC(c2ccc(F)cc2C)=O)C(O)C1 N1(C(=O)CC23CCCC2C3)CCCC(CC(=O)NOCC2CCC2)CC1 CCCCCC(C)CC(=O)NC1(CF)CCN(C(c2cc(C)c(N)cc2Cl)=O)C1 Cn1cnc2nc(C(N3CCC4C(NC(c5ccccc5Br)=O)C34)=O)ccc12 N1(C(c2c(CC)ccc(F)c2)=O)CC(C2CN(C(=O)C(F)(F)CC)C2)C1 N1(C(c2cncc(C#C)c2)=O)CC2CN(C(=O)C(COC)OCC)CC2(C)C1 N#Cc1ccc(COC(=O)C(O)Cc2ccccc2Br)cc1 c1(C(=O)NC2CC(C)CN(C(c3nn[nH]c3Cl)=O)C2)ccc2c(c1)C(=O)NC2=O C1(NC(CCC)=O)CN(C(c2cc([N+](=O)[O-])nn2C)=O)CC12CCC2 Cn1cnc2cccc(C(=O)NC34CCCC3CN(C(=O)CCCC(N)=O)C4)c12 C1(NC(C2N(C(C)C)C(=O)COC2)=O)CCCN(C(C2(C)CCOC2)=O)CCC1 c1(NC(C2(CCl)CCN(OC)CC2)=O)cc2scc(Br)c2[nH]1 C1(NC(c2cncc(OC)c2)=O)CC2(C1)CC(NC(C1CCCC(OC)C1)=O)C2 C1(C(=O)NCCCC(C)NC(c2ccco2)=O)CNC(=O)C(C)(C)C1 C1(NC(c2cccc(CC)n2)=O)CN(C(c2cc[nH]c2C)=O)Cc2ccnn2C1 C1(C(=O)NC(CCC(=C)C)C)CC2CN(C(c3nc(Cl)oc3C)=O)CC2C1 Cc1ccnnc1C(=O)NCC1(C(=O)N(C)CC2CCC(C)CC2)CCCC1 c1(C(=O)NC2CC(F)(CNC(Cc3n(C)c(S)nn3)=O)C2)cc2n(n1)CCOC2 C1(C(=O)NC2CCC(O)CC2)CCC(O)CN1C(=O)C1CC1 N1(C(C(N2CCCN(C(=O)NC)CC2)=O)=O)CCCc2sc(C(=O)OC)cc2C1 c1(C(=O)NC2C3CC(O)C2N(C(c2ccsc2)=O)C3)cc2cc(Cl)ccc2o1 C1(C(N2C(C(=O)NCc3cncc(O)c3)C3CCC2C3)=O)CC(=O)NC(=O)C1 C(=O)(C(CC(N)=O)NC(=O)C=C(C1CC1)C1CC1)NC(C=C)(C)C C#CCC(C)(C(=O)N1CC(C)CC(O)C1)NC(=O)C(F)CCCC N1(C(C2C(OCC)C2)=O)CCC(O)(C(C)NC(c2cc(Cl)ccc2N)=O)CC1 C(=O)(CCN=c1[nH]ccs1)N1CCCC(CNC(C(C)OCC2CC2)=O)C1 CCC(CC)C(=O)NCC=CCNC(c1conc1C1CCC1)=O c1(OC)ccnc(Oc2ccccc2F)c1.c1(OC(=O)NC2CC(N)C2)n[nH]cc1F C#Cc1ccc(C(=O)NC2CN(C(c3ccc(SC)o3)=O)CC2C2CC2)c(C)c1 C(=O)(C1=CC2CC=CCC12)NC1(CNC(C(C)(C)n2cc(Cl)cn2)=O)CCC1 N1(C(C2N(C(c3ccnc(C)n3)=O)CC(O)CC2)=O)CCC2(CCOC2)CC1 c1(C(N2CC(CNC(=O)C=Cc3cccs3)C3C2C3)=O)c(F)c(F)cc(F)c1F C(=O)(C(CC(C)C)C(N)=O)Nc1nc(=NCC2CCCC(C(=O)OC)C2)s[nH]1 C1(NC(c2cncc(CC)c2)=O)CCN(C(=O)CCn2ccnc2)CCC1CO N1(C(CCC)=O)CCCC(CCNC(=O)CC2CC(=O)NC2=O)C1 C#CC1(C(=O)NC(c2cn(C)nn2)(C)C)CCN(C(=O)CC2(COC)CC2)C1 N1(OC(=O)C=CCOCc2ccco2)CCC(c2ccc(F)cc2)OC1=O C1(C(=O)NCCOCCNC(C(C)=C(C)C)=O)CCc2nc(C(C)C)cn2C1 C1(NC(C(CC)NC)=O)COC2CN(C(c3cccc(Br)c3F)=O)CC12 C(=O)(C(C)(O)CCC)NC1CN(C(Cc2ccc(CCC)cc2)=O)CC1C(F)F c1(C(=O)NC(C)CCCNC(=O)C=C2CCN(C)C2)cc(C(F)(F)F)n(C(F)F)n1 C(=O)(C(C)S)N.C(C(COCCOCCOC(C)C)NC)CC c1(-c2cn(C(C)C(=O)N3CC(N4CCC(O)C4)C3)nn2)cc(F)c(Cl)c(Cl)c1 CC1CCCN(C(=O)C(=O)NCc2ncc(C(C)C)s2)CC1 C1(C(NOCC(=O)NC2CCCC2O)=O)(CC=C)CCCC1 c1(C(C)SCC)ccccc1NC(c1cc(CC(C)C)on1)=O c1(C(N2CC(SC)C(NC(C3CCCC3(F)F)=O)C2)=O)cc2cc[nH]c(=O)c2s1 c1(NC(C2C(C)(C)CCNC2)=O)ccc2cc(S(N)(=O)=O)ccc2c1 CC1=NOC(=O)C1CC(=O)NC1CC(n2cnnc2)C1 c1(C(=O)NC2C(CNC(C3CC(OC)C3)=O)COC2)ccc(Cl)c(Cl)c1 N1(CC(=O)N(C)CCc2ccc(Cl)cc2)CCc2c(cccc2S(N)(=O)=O)C1 C1(C(=O)NC2(CNC(C(C)(C)OC(C)=O)=O)CCCC2)CC2(CCC2)C1 CC(C)C(C)C(CNC(=O)OC(C)(C)C)C(=O)N1CC2(C)CC1CCO2 c1(C(=O)NCC2C(C)CCN(C(C(CC)(C)O)=O)C2)ccc(C)c2c1CCCN2 Cc1ccc(C)c(C(N2CCOC(CN(C)C(C3CCOC3C3CC3)=O)C2)=O)c1 N1(C(=O)OC(C)(C)C)C2CCC1CC(NCCN1CCC(O)(C(=O)O)CC1)C2 Cc1cc(C(=O)NC(C)(C)CCCNC(=O)CCC(C)c2ccccc2)[nH]c1C C1(N(C(C2CC=C(C)CC2)=O)C)CCC2CN(C(C3CC3(C)C)=O)CC12 N1(CC2(CC)CCC2)CCCC(C)(C(=O)NC(C)CC2CC2(C)C)C1 c1(C(=O)NC2(CCC(=O)NC3(C=C)CCOCC3)CCC2)cccc2ccnn12 C12CCCC1CNC2=O.C1(CNC(C(C)=CC2CC2)=O)C=CCCC1 c1(CCC)cc(C(N2CCC(N(C(=O)C(C3CCOCC3)F)CC)C2)=O)ccn1 C1(O)(CC#C)CCN(C(=O)C(C)(C)CCNC(=O)CCSC)CC1 C(=O)(C(CNC(c1ncc[nH]1)=O)CC1CCCC1)N(CC(C)CO)C c1(CC)ccc(F)cc1C(N1CC(O)(C(C)NC(C2CC2C(C)O)=O)C1)=O C1(NC(CC(C)=C(C)C)=O)C(CNC(=O)CS(C)(=O)=O)CCC12CCC2 N1(C(c2nnc(C)s2)=O)CCCCC1CN(C(=O)Cn1cnc(C(N)=O)n1)C C(=O)(C(C)(C)C(=O)NC1CC2(NC(=O)C(C)OCCO)COC1C2)NCCOC O=C(NNc1cccc(F)c1Cl)NCCOc1ccc(Br)cc1C(F)(F)F c1(NC)ccc(C(N2CCC(N(C)C(c3ccc(C)c(F)c3)=O)CC2)=O)cc1F C(=O)(CC(O)C(C)(C)C)NCC1OCCN(C(CN(C(COC)=O)C)=O)C1 C(N=c1[nH]c(-c2ccccc2N)cs1)c1c(C)cccn1 C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(C)NC(c2ncn(C(C)C)c2)=O)C1 c1(C(C)C)nc(CC(=O)NC(c2ccco2)=O)no1.C1(=O)C(C)O1 C(C(CCC)OC)NC(C(c1ccco1)NCC1(CCC=C)CC1)=O c1(C(N(CCC2N(C(CCCC)=O)CCCC2)C)=O)ccc2cc(C)oc2c1 CC1CCCN(C(c2cnoc2C2CC2)=O)C1CNC(=O)CCC(N)=O CC1OC2CCC1(NC(C1(NC(C3CN4CCC3CC4)=O)CSC1)=O)C2 C(C1=NOC2CN(C(=O)CCc3cncn3C)CC12)NC(Cn1c(C)ccn1)=O c1(OC)ccc(NCCCN(C)C(c2ccccc2)=O)cc1F c1(C(=O)NCCNC(Cc2scc(C(=O)OC)c2)=O)cc(O)c2c(cnn2C)c1 C1(CNC(C(C2CCCOC2)OC)=O)CCN(C(C2(F)CCOC2)=O)C1 CC(C)CC(=O)N1CCC(C(NC2CCCc3n[nH]cc32)=O)O1 N1(C(=O)OC(C)(C)C)CCCC2CN(CSc3ccc(Cl)cc3Cl)CCCC12 C1(OC)CC(NC(=O)CC2CC3C=CC2CC3)CN(C(c2cc(O)ccc2Cl)=O)C1 c1(C(C(=O)NC(CNC(c2cc(C(C)=O)sc2)=O)C)(F)F)cccc(C)c1 C(C)(CS(N)(=O)=O)NC(c1ccc(F)cc1)c1n(CCCOC)nnn1 C(=O)(C1=CS(=O)CCC1)NC1C(NC(CCCCCOCC)=O)CCCC1 N1(C(C2CC2)=O)CCCC(C(N2CCC(N3CCCCC3)C2)=O)C1.N1CCCC1 Cc1ccc(Cc2nc(-c3ccoc3)nn2C2CCC(C)C2)cc1Br Cn1c(Nc2cc(-c3cccc(Sc4ccccc4)c3)ccn2)ccc1C#N N12CCN(CC1)CCC(=O)N2C1CN(C(=O)CO)CC1C.CC(C)(C)C1CC1 CC(C)CC(CCc1ccccc1)C(=O)NCCNC(C12CCCN(CCC1)C2)=O N1(Cc2scc(C(=O)OC)c2)CCOC2C1C2(F)F Nc1ccc(Cl)c(C(=O)NC2CC2CNC(c2ccnnc2S)=O)c1 N1(C(C2C(C=C)C2)=O)CCN(C(c2ccc(CC)s2)=O)CC1Cn1cc(Cl)cn1 CCCCCCCC(F)C(=O)NCCCN(C)C(c1ccc(CO)s1)=O C(=O)(CCC(=O)NC1(C)CCN(C(C2(C(N)=O)CCC2)=O)C1)NCCC c1(C(=O)O)ccc(NS(=O)(=O)Cc2cc(Br)ccc2Br)cc1Br c1(CC)onc(C)c1C(=O)NC(C1(CNC(c2[nH]c(C)nc2C)=O)CC1)C c1(N(C2CCC(CSC)CC2)c2ccccc2)ncnc(NC2CC2(Cl)Cl)c1C CCCN=C(NCC1C2(CC2)C12CC2)NC1CCN(c2ccccn2)C1 c1(C(=O)NCC2(CNC(C(F)=CCC)=O)CC2)ccccc1OC C1(OCC(=O)N(CCOCCC(=O)OC)CCO)CCN(C)CC1.C(C(F)F)O C1(CNC(=O)C2=CCCC2)CCC2(CN(C(c3cncc(Cl)c3Cl)=O)C2)O1 Cc1cc(NC(=O)C(C)N(C(=O)C=Cc2ccncn2)C)cc(C#N)c1 c1(CC(=O)C(N2CCC(C)(CN)C2)=O)c[nH]c2ccccc12.N C1(CNC(C=C(C)C)=O)CCN(C(C2CC3(CSC3)C2)=O)C12CC2 C1(C(N2CC(C(C)C)C2)=O)COCCN1C(c1cccc(Cl)c1)=O c1(C(=O)NCCCNC(C(CCC)C#N)=O)ccc2cc(F)ccc2n1 c1(C(C)C)ccc(C(=O)NC(C)CN(C)C(C2(C(N)=O)CCC2)=O)c(O)c1 N1(C(C(C)=CC)=O)CCC2(CCOCC2)C(CNC(=O)CC2CSCCS2)C1 C1(C)(CC(=O)NCC(c2ccncc2)C)CCN(C(=O)CCn2ccnc2)C1 C1(NC(=O)Nc2[nH]ccc2COC)CN(C(C2(OCC)CC2)=O)C2(CCOC2)C1 N12CCCC1C(=O)NCCN2C.C1(C(=O)N)CCCN1S(C)(=O)=O.C1(CC)(C)CC1 N1(C(c2[nH]ccc(=N)n2)=O)CCCCC(CC(=O)N(CC2CC2)CC2CC2)C1 c1(C(N2CC(CNC(C=C(C)c3ccco3)=O)C(C)C2)=O)c[nH]c2nccc-2c1 CCC(CC(=O)NC1CC2CCC1N(C(=O)CS(=O)(=O)C1CC1)C2)C(C)(C)C C(=O)(C(C)(C)CC(C)(C)C)NCC(CN(C(C1N(C(CCC)=O)CCC1)=O)C)O C1(CNC(CC2N(C(CC(CC)SC)=O)CC2)=O)OC(=O)CC1(C)C N1(CC(C)NC(CC(C)F)=O)CCN(C(=O)CCCn2cccn2)CC1 C1(CN(S(=O)(=O)CCOC(C)(C)C)CC)CCCC1(C)C N1(C(C2CC(OC)C2)=O)CCC2(CCN(C(=O)Cc3ccc(C)s3)C2)C1 C1(CNC(C(CCC)=CCC)=O)CCCCN(C(C2Cc3nncn3C2)=O)C1 Cc1nnc2n1CCC(C(=O)NCCN(C(=O)C=CC1CCCO1)C1CC1)C2 c1(N(C)C)ncc2c(n1)CCN(c1[nH]c(=N)nc3c1cnn3C)C2 CC1CCCC1(C(=O)N(C)CCC1CCCO1)NC(c1cnn(C)n1)=O N1(C(c2c(C(C)C)ncs2)=O)CC2C(CNC(=O)C(F)n3ccnc3)C2C1 C(C(C)(O)CNC(=O)CCc1ccnn1C)NC(CCC1CC(C)C1)=O CC1CCC(c2nc(CCO)nn2-c2ccnc3ccccc23)CC1(C)C N1(C(CCC#C)=O)CCC(C2CCN(C(C34CCC(OC)C3CC4)=O)CC2)CC1 CCC(C)(CNC(c1cc(C#N)n(C)n1)=O)C(=O)NC(C)C(C)(C)C C1(NC(C(CCC=C)(C)C)=O)CC2CCC(C1C)N2C(=O)OC(C)(C)C c1(CN2CC3CN(C(C4(c5ccccn5)CC4)=O)CC32)cc(F)c(Cl)cc1F c1(C(=O)NC(CNC(c2ccc(CC)o2)=O)C)csc([N+](=O)[O-])c1 Cn1cc(CCC(=O)NCC2CCC2NC(C2(C(F)(F)F)CCO2)=O)cn1 N1(C(CCOCCOCC)=O)CC(NC(=O)C=C2CC2)C2(CCC2)C1 C1(C(N2CCC3(CSC3)C2)=O)(CC)CCCN(C(=O)C(C)C(F)(F)F)C1 CC(C)C(O)CC(=O)NCCC1(O)CN(C(=O)COCC(c2ccccc2)C)C1 CN1CCC(C(=O)NC(CO)C(N)=O)(NC(C2CC(C)(O)C2)=O)C1 C1(C(=O)NCc2ccc(SC)cc2)CC2CCC1N(C(c1cc(O)n(C)n1)=O)C2 C(C)(C)(CCCNC(=O)Cc1cnoc1)NC(c1ccc(NC(C)=O)s1)=O CCC(C)(C(=O)NC(CNC(C1(C)CCSCC1)=O)C(C)C)OC N1(C(Cn2ncc(S(C)(=O)=O)c2)=O)CC2CS(=O)(=O)CC2C1.c1(N)ccccc1 C1(NC(C2CCC(CC)O2)=O)CN(C(c2ccoc2C(C)C)=O)CCC12CCC2 N1(C(c2n(CCC)ncc2)C(=O)NCCOC)CCOc2ccc(F)cc2C1 CCC(CC)(CC)C(=O)N(CCNC(c1cc2ncccc2o1)=O)C1CC1 C(=O)(C1Cc2ccccc21)N(C)CC1CCN(C(=O)Cc2cn(C)nc2Cl)C1 S(=O)(=O)(c1sccc1C#N)N1CCCN(c2c(C)cccc2Cl)CC1 N1(C(C(C)(C)CSc2ccccc2)=O)CC(C(=O)NOC2CCC2)CC(F)C1 CC(C)(CC1CC1)C(=O)NCCC1CCN(C(=O)CCC2CCCC(=O)N2)CC1 c1(NC(=O)NCC2CC2C(F)(F)F)ccncc1F C1(C(=O)NCC2CC(OC)CN2C(=O)C#CC(=O)N(C)C)Cc2ccc(C)cc2S1 CC1=NOC(C)(C(=O)NCC2(NC(c3c[nH]nc3Br)=O)CCOC2)C1 N1(CC2CCCC(CF)C2)CC(=O)N(Cc2cc(-c3ccccc3)n[nH]2)C1=O C1(CNC(C(C)NC(=O)OCC)=O)CCC(NC(c2cnc(C(F)(F)F)s2)=O)C1.CC C(C(=O)N=c1ccn(C(C)CC)[nH]1)C1(NC(C(CCC)CCC)=O)CCCC1 N1(C(C(C)(C)c2ccns2)=O)CCC(NC(=O)CC(F)(F)F)CC1C1CC1 C1(C(=O)OC(C)(C)C)CCN(C(c2ccc(SC(F)F)cc2)=O)C12CCCC2 CCCCCC(C)(C)CNC(C1COC2(C1)CN(C(=O)C=CCCCCC)C2)=O C1(C(=O)NC(CCSC)C)CN(C(=O)CC2CCCCCCC2)C(C)(C)C1 C1(CN(C)C(C2CC23CCC3)=O)CCCN1C(c1cc(Cl)c[nH]1)=O c1(C(N2CCC(C(=O)NC3C=C(C)CCC3)CC2)=O)cc(O)ccc1F CCCC(CCC)C(=O)N(CC(C)C(N1CC(CO)CC(C)(C)C1)=O)C N1(C(C(C)NC(c2c(C)onc2)=O)=O)CCOC(CNC(=O)C(C)(C)O)C1 c1(CC)ccc(N)c(C(N2CC(CNC(=O)CC(C)(C)SC)C(O)C2)=O)c1 C=C(C)c1ccccc1NC(=O)CCC(C)NC(=O)CCc1ccco1 N1(C(CCOCC)=O)CC(C2CCN(C(c3ccc4c[nH]nc4c3)=O)CC2)C1 C#Cc1cnc(C(=O)NCC(C)N(C(=O)C(CC)NC(C)=O)CC)c(C)c1 c1(C(N(C2CCN(C(CC(C=C)(C)O)=O)C2)C)=O)ccc2c(c1)CC(C)(C)O2 c1(CC)ccc(F)cc1NC(=O)CCNc1cccc(O)c1OC O=C1CCC(C(=O)NCC2(NC(=O)C=CC3CCOC3)CC2)N1 C(=O)(C(C)(C)C(C)NC(=O)CCc1nccs1)NC1(CCOC)CCC1 CCCCC(O)CC(=O)NC1CCC1OC c1(C(C)C)nc(NCC2CC3(CC3)C2)cc(=NC2CCOc3c(Cl)cccc32)[nH]1 C1(C(=O)OCC)CC12CCN(C(=O)Oc1cncc(F)c1)C2 C1(C(=O)Nc2nc(Cl)cs2)CN(C(=O)CC=C(Cl)Cl)CC1c1ccccc1 C1(NC(C(CCSC)NC(N)=O)=O)CC2CCC1N2C(=O)C1=CSCS1 c1(CC(=O)N(CCCNC(C2(F)CCOC2)=O)CCO)ccc2c(c1)CCOC2 N1(C(COCCC)=O)CC2CCN(C(c3cccc(C(N)=O)c3F)=O)CCC2C1 N1(OC(=O)CCNC(c2cccnc2)=O)CC2CC(C1)CS(=O)(=O)C2 c1(C(=O)NCCC2CN(C(C3(C#N)CC4CC4C3)=O)C2)nc2c(s1)COCC2 c1(C(=O)NC(CNC(c2ccc(CCC)cc2)=O)CO)ccnc(Cl)c1F C(=O)(C(CCC1CCCOC1)N1CCSCC1C)NC c1(C(=O)NC(CNC(C2(SC)CCC2)=O)C)cnn(CCO)c1N N12CCC(C)(C1)NCC2=O.N1(CCC(C)SC)CCOCC1 N#Cc1cccc(O)c1NC(c1ccnc2ncccc12)=O c1(C(=O)NC(CN(C(C(C2CC2)SC)=O)C)C)[nH]cc2c1CCCC2 Nc1ccc(N2CCNCC2)c(C(=O)NCCCC2CCCC(F)(F)C2)c1 c1(NC(C(c2scc(COC)c2)N(C)Cc2ncco2)=O)cccc([N+](=O)[O-])c1 CCCCC(F)C(=O)N1CCCC(C(N2CC(C(N)=O)(OC)C2)=O)CC1 C(C(O)CO)NC(C(=O)N(CCCO)CCC)=O N1(C(COC(C)=O)=O)CC23CCCC2(C1)CN(C(c1ccc2c(c1)C(=O)NC2)=O)C3 C1(C2CCC2)(CN(C(=O)CC2COC(C)(C)C2)C)CC1.C1(=O)CC2(CC2)CN1 C1(C(=O)NCC23OCC(CNC(=O)Nc4ccc[nH]4)(C2)C3)CCC(C2CC2)CC1 N1(C(CN(C(CSCCC)=O)C)=O)CCCN(Cc2ccccc2Cl)CC1 N1(C(=O)NC)CCCC1C(=O)NC1(CNC(C2(O)CCOC2)=O)CC1 c1(CNC(=O)NCC=CCO)ccc(OC(F)F)cc1F C1(C2CC2)(C(N(CC)CC2CCN(C(c3coc(Cl)n3)=O)CC2)=O)CCOCC1 Cc1ccc(C)c(C(=O)NC2CC3(C2)CN(C(C24CCCC2C4(F)F)=O)C3)c1N N1(C(C(COC)N(C)C)=O)CCC(N(C)C(c2ccc(N(C)C)nc2)=O)CC1 C(=O)(C(C)(C)C(F)(F)F)N1CC(CNC(c2ccc(CC)s2)=O)OCC1 CC1CCN(C(C2C=CCC2)=O)CC1CNC(=O)Cc1cc(C2CC2)n(C)n1 C#Cc1ccc(NC(=O)C(CC)N(C2CC2)CC)cc1.C1C(O)CN1 c1(CC)noc(C(=O)NCC2(F)CC(CNC(C3(C)CCOC3)=O)C2)c1C n1(CC)nccc1C(=O)NC(C1(O)CN(C(=O)C(N2CCNC2=O)C)C1)C CS(=O)c1ccccc1-c1cn(C2CC3(C2)C(C(=O)O)C3(F)F)nn1 c1(CC)cccc(F)c1C(=O)NCCOCCCNC(=O)C(C)Cn1ccnc1 c1(C(N(C2CCN(C(C3C(CC)C3)=O)C2)C)=O)ccc2c(c1)C(=O)NCC2 c1(C(=O)NC2(CC)CCOCC2)cc(O)nc(OC)n1 N1(C(Cc2cc(C)ns2)=O)CCN(C)CC1C(=O)NCC(C)N(C)C c1(CC)occ(C)c1C(=O)NC(CCN(C)C)C(C)C c1(C(N2CC(CC)N(Cc3cc(Br)c[nH]3)CC2)=O)cc(F)c(F)cc1Br C1(C(N(CCNC(CCOCC#C)=O)CCOC)=O)C(C(F)(F)F)C1(C)C N1(C(C2C(CC)OCC2)=O)CCC(NC(c2cn(C)c(C(F)F)n2)=O)C(C)(C)C1 c1(NC(C(c2ccccc2Cl)SC)=O)nc2ccsc2s1 c1(CC)cc(C(=O)NCC2CC(C)(C)CN2C(c2cscc2OC)=O)c(C)nn1 CN1CCN(C)C(C(N2CCN(CC3CCN(C(=O)C(N)=O)CC3)CC2)=O)C1 c1(C(=O)OC)cc2c(N(C)C(c3cc(C)c(Cl)c(C)c3)=O)cccc2s1 c1(C(N(CCC)CCNC(=O)Cc2ccc(O)cc2Cl)=O)ccc2nnnn2c1 N1(C(C2(C=C)CCC2)=O)CCOC(C2CN(C(C3CC=CCC3C)=O)C2)C1 C(CNC(C1Cc2nccn2C1)=O)(CC(F)(F)F)NC(C=CC(C)C)=O c1(-c2c(OC(C)=O)cccc2)c(C(N2CCC(F)CC2)=O)nn2c1CCCC2 C1(CCCC)CCCN(C(C2CC(CNC(c3cccc(NC)n3)=O)C2)=O)C1 CC1(C(=O)NCC2C3CN(C(c4cocn4)=O)CC23)CCCCC1(F)F C=CCC(C)(C)CC(=O)N1CC2CC(NC(=O)Cn3cnc(C(N)=O)n3)C1C2 N1(CC)CC2(CSC2)C1.c12cnc(s1)C1CN2C1.n12cc(nn1)COC2=O N12CCc3nc(sc3C1)CC=CC2=O.C(=O)CCC(C)(C)F.CC(C)(C)OCC=C C(=O)(C1=COCCO1)NCC(C)CNC(C1CCOC1C(F)(F)F)=O C1(NC(CCCCC)=O)CCC2(CC1)CCN(C(=O)C#CC1(C)CCCCO1)C2 c1(C(C(=O)Nc2ccccc2Cl)N(C(CSC)(C)C)C)ccc(C)cc1F c1(C(N2CC(CCNC(C3CCC4CC4CC3)=O)OCC2)=O)n[nH]c2c1CCC2 Cc1ccc2c(cnn2C)c1-c1cc(C(=O)Nc2cc(F)cc(F)c2Cl)n[nH]1 C(=O)(C(CC(F)F)NC(c1csc(=N)[nH]1)=O)N1C(C=C)CC1 C1(C(N(CC(C)NC(=O)CCc2cncn2C)C)=O)C=CCCC1 S(=O)(=O)(c1cc(F)cc(Br)c1)NC1CCCN(S(CC(C)C)(=O)=O)C1 c1(C(N2CCC(NC(C3(Cl)C(C)(C)C3)=O)C2)=O)cccc(Cl)c1O C1(NC(=O)Nc2ccc(CC3(C(F)(F)F)CC=CC3)cc2)CCC2COCC2O1 C(C(C(=O)NC1CCCC2(C1)N=N2)C(C)C)NC(c1cncc(C)c1)=O C1(C(N(C2CCCC2)CCCNC(=O)CC2CCC2)=O)C2C3CCC(C3)C12 C12(C(=O)NC(C)CNC(=O)C(C)(C)c3ccnn3C)CC1COC21CCC1 C#CCC(C)(CC)C(=O)N1CCOCC(CNC(C2CC3(C2)CC(C#N)C3)=O)C1 CCCCCCCCCC(=O)NC1CC2CC(C1)N(C(C13COC(C1)C3)=O)C2 c1(C(=O)NC2C(NC(CCN(CCC)C)=O)C2)c[nH]c(Br)c1 Nc1ccc2[nH]c(C(=O)NC(C3CCCC3)CNC(=O)C(=O)N3CC3)cc2c1 c1(C(=O)NC2CCN(C(CC(C)n3cccn3)=O)CC2F)[nH]nc([N+](=O)[O-])c1Cl C(CC(C)(C)CN=c1[nH]c(=NC2CCS(=O)C2)[nH]c2c(F)cccc12)OC Cc1[nH]nc2ccc(C(=O)NC3C4CC3N(C(C3(COC(C)C)CC3)=O)C4)cc12 C1(C(N2C(C)(CC(=O)NCC(N3CCOCC3)C)CCC2)=O)CC2CC1C1CC21 CC1(C)C(NC(=O)OC(C)(C)C)CCCN1C(C1CCC2CC1C2(C)C)=O N1(C(CC#C)=O)CC(NC(c2cc3cccnc3s2)=O)CC(F)(F)C1 C(=O)(C(C)CCS(C)(=O)=O)N1CCN(C(C2N(C(CCC)=O)CCC2)=O)CC1C Cc1nc2ccc(CNC(c3cnc4ncccn34)=O)cc2[nH]1 Cc1ccc(C)n1CCNC(=O)Cc1cscc1Br c1(OC)ccc(C(N2CC(=O)NC(C)C2)=O)c(Br)c1OC.C123CC(C1)(C2)C(=O)N3 c1(NCC2CC(NC(=O)CSc3nc[nH]n3)C2)nc2cc(F)ccc2s1 c1(C(=O)NC2(CF)CN(C(c3cnc(=N)[nH]c3)=O)C2)coc2cc(O)ccc12 CC(C)CC(C(=O)NCCC1(CNC(C2(F)CC2)=O)CC1)N(C)C.N(C)(C)C c1(OC)cc(NC2CC2C(=O)NCCC2=CCCCC2)nc(S(C)(=O)=O)n1 c1(C(C(=O)Oc2ccc(OC)cc2OC)C)ccc([N+](=O)[O-])cc1F Cc1ccc2oc(N3CCC(=CCNC(c4cc(CO)c(C)o4)=O)CC3)nc2c1 Cc1cc(Cl)ncc1CC(=O)NC(C)C(CO)NC(c1cc(F)n(C)n1)=O CC1(C)COC(C(=O)Nc2cccc(C(=O)NCCC(F)(F)F)c2)C1 c1(C(N(CC(CC)NC(C2(OCC)CCSCC2)=O)C)=O)c(C)ncnc1O C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1cnoc1)NCCC1CCN(C)C1 C=Cn1ncc(C(=O)NCC2(C(=O)N(C(C)CO)C)CC3(CC3)C2)c1N N1(CCNC(C2(F)CCC2)=O)CCCN(C(C2(F)CCCOC2)=O)CC1 C(CCC(=O)N1C(C(=O)NCC2(C3CC3)CC2)CC1C)=CC(C)C C12(c3ccccc3)CCC(C1)NC(=O)C(C)NS(=O)(=O)C2.C1(CSCC)CC1 c1(C(=O)NC(C)CNC(=O)CC2CN(CC(F)(F)F)C2)ccc2nccn2c1 N1(C(c2cccc(OCC(C)C)c2)=O)CCN(C(=O)CN(C)C2CC2)C(CF)C1 c1(OC(C(=O)NCC(=O)OC)C)cc(Br)ccc1C(=O)OC n1(-c2n(C)nnc2)nc(-c2ccc(Cl)cc2)nc1Cc1cc[nH]n1 c1(C(N2C(CNC(C3CC4(CCCCC4)C3)=O)C=CC2)=O)cn2cccnc2n1 C1(NC(C(c2cnn(C)c2)C)=O)(CO)CN(C(=O)C(C)(C)NC(=O)OC(C)(C)C)C1 C(CCCCN=[N+]=[N-])NC(CC(C)CNC(C1C2COCC12)=O)=O C12(OCCNC(=O)Cc3ccno3)CCC(CC1)C2 C1(C(=O)NCC2N(C(C3(CN(C)C)CC3)=O)CC2)CC(c2cccnc2)=NO1 S(=O)(=O)(c1ccc(C)c(C(N2CCC(COc3cccnc3Br)CC2)=O)c1)NC C1(CNC(C2CSCCS2)=O)CCN(C(C23CCC(F)(CC2)C3)=O)C12CC2 N1(C(CC(CNC(=O)C=Cc2ccsc2)OC)=O)CCC(F)(F)CC1 C1(C(N2CC(C)OC(C)(C(F)F)C2)C(=O)NC(CC)C)C2(CCC2)C12CCC2 c1(C(=O)NCCC2(C(N(C)CC3(C)CC3(F)F)=O)CCC2)cnn2c1OCC2 C1(NC(C(CCC)O)=O)(COC)CCN(C(C2CCC(=O)N(C)C2)=O)CC1 C(CCC(C(=O)NC(C1(O)CCC1)C)NC(c1cnc(O)c(F)c1)=O)OC Cc1cc(Cl)c(C(=O)NCCC23CCC(C2)N(C(=O)C(=O)NC(C)C)C3)cc1F c1(CCC(=O)N(CC(CC)NC(=O)C(CCSC)OC)C)ccccc1F c1(CC)nc2ccc(Cl)cn2c1C(=O)NC(C)CNC(c1cocn1)=O C12(CCNC(Cc3c(C)noc3C)=O)CCC1CN(C(c1ncncc1Cl)=O)C2 C1(c2cccc(OC)c2)CN(C(=O)C=CBr)CCN1C(=O)CN1CCC(C)(C)C1 CCC(CC)CCCNC(=O)CC1(NC(=O)C(C#N)C(C)C)CC1 N1(C(C(CC(C)C)N(C)C)=O)CC(F)(F)CC1(C)CNC(=O)CCN1CCOCC1 c1(C(N(C(C)CNC(=O)CCCOC(C)(C)C)CC)=O)cc(C(C)=O)cs1 c1(C(=O)NCCOCCN(C(=O)COCC2CCCO2)C)nccc2ncccc12 c1(C(N(C2CN(C(C3C(CC)OCC3)=O)C2)C)=O)cc(F)c(O)c(Cl)c1 c1(C(C)C(=O)NC2CC(CNC(C34CCC(C3)C4)=O)C2)cccc(F)c1 C(=O)(C1=COCCC1)N1CC2C(CNC(c3n[nH]cc3C3CCC3)=O)(C2)C1 c1(SCC(=O)NCC(CNC(=O)C(CO)N(C)C)OC)ccc2nn[nH]c2c1 c1(C(N(CCO)Cc2cn(C3CC(C(N)=O)C3)nn2)=O)noc2c1CCCCC2 N1(C(c2c(SC)cccc2)=O)CCN(C(=O)CC2CCOC(C)(C)C2)C2CCC12 CC(C)CCC(O)C(=O)NCCC1CC(NC(C2CCC(C)(C)C2)=O)C1 c1(CC(=O)N(CCCNC(CCC(C)SC)=O)C)nc2ncccn2n1 N1(C(Cc2c(C)cco2)=O)CC(C)(C)CC1CNC(=O)CN(C)C c1(C(=O)NC2CCN(C(c3c(C)sc(Cl)n3)=O)CC2F)cnc2[nH]ccc2n1 Cn1cncc(C(=O)NC2(CCNC(=O)CC3CCCC34CC4)CCC2)c1=O N1(C(CSCCOC)=O)CC(NC(C2CCCC(C(C)(C)C)C2)=O)C(N=[N+]=[N-])C1 CCCC(C(=O)NC1CCCCC1NC(=O)C(c1ccc(C)cc1)(F)F)N(C)C CC(C)(C)C(C#N)C(=O)NC12CC(C(=O)NCCN3CC=CCC3)(C1)C2 c1(C(=O)NC2(CCOC)CCN(C(=O)CCC(F)F)C2)nccc2cc[nH]c12 C1(NC(CC(=O)NCC)=O)CC2CCCC(C1)N2C(c1ccnc(F)c1O)=O c1(C(C(=O)NCCOC)CN2CC(SC)CCC2C)cccc(F)c1F CC(C)(CNC(C1CC(O)CN1C(=O)CC1CC(=O)NC1=O)=O)C(F)(F)F N1(C(CC2COCC(C)O2)=O)CCCC(C(N2CC(F)(C3CC3)C2)=O)CC1 CN1CC=CCC1CC(=O)NCCOC1CCN(C(c2c[nH]cc2Br)=O)CC1 c1(C(N(C)C)=O)ccc(C(F)(F)F)cc1N.c12csc(n1)CNC2=O C(=O)(CCCN(C)N=O)N(C)CC1CCCN(C(C2N(CC)CC2)=O)C1 CC1(C)CCN(C(=O)C2=CCCS2)CC1NC(C1CC1F)=O C1(NC(=O)COCCCF)CN(C(c2cncc(CO)c2)=O)CC12CCC2 C1(C(N(CC(C)NC(c2cc(O)nc(O)c2)=O)C)=O)CC2(CCC(F)(F)CC2)C1 CC1CC1N=c1nc2c(ncn2C)c(NCCOc2ccc(Br)cc2)[nH]1 c1(C(=O)NC(C(C)NC(C(CC)(CC)CC)=O)C)nc(SC)n2ccccc12 CCC(Cc1cn(-c2ncc(C(=O)OC)cn2)nn1)C(=O)O C1(NC(Cc2ccc(C(C)=O)[nH]2)=O)COCCN(C(c2cnc(C3CC3)s2)=O)C1 C1(CN(C(C2(OC)CCSC2)=O)C)C2CN(C(c3cccnc3C(F)F)=O)CC12 c1(OC(C(=O)NCCN(C(CC(C=C)C)=O)C)C)ccc(F)cc1Cl C1(CCNC(C2CCC2(F)F)=O)CCN(C(c2nocc2Cl)=O)C1 N1(C(=O)NCC(c2ccccc2)C)CC(C)C(NC(=O)NC(C)(C)C)C(C)C1 C12(CNC(CCNS(CC)(=O)=O)=O)CCC(CN(C(=O)C(C)(C)CCC#N)C1)C2 N1(C(c2ccc(CC)[nH]2)=O)C2CCC1C(F)C(NC(=O)CC1CCCCO1)C2 N1(C(c2cc(CC)sn2)=O)CCC(C(=O)NCc2cn(C)nn2)C(O)C1 C(CC(C(=O)N(C)CCc1cnn(C)c1)OC)NC(C1C(=C)C1)=O N1(C(Cc2n(C)ncc2Cl)=O)CCN(C(=O)COC2CC2)C(CCO)C1 c1(C(CN(C(C)C)C(c2csnc2Br)=O)O)ccccc1 C1(COC)CN(C(c2scnc2Cl)=O)CCN1C(c1ccc(CN(C)C)o1)=O CC1(F)COCCN(C(C2CCCCCCN2C(C2CC3C(C2)C3(F)F)=O)=O)C1 c1(C(C)NC(=O)N(CC2CC2)CC2CC2)cccs1 N1(C(c2c(C)ccc(C(N)=O)c2)=O)CCC(C)(C)C(NC(=O)CCCC2CC2)C1 N1(C(C=CC=CC)=O)CC2CCCC2(CNC(=O)Cc2ccc(C)cc2)C1 c1(C(N2CC(CC(=O)Nc3ccc(C)cc3)(OC)C2)=O)ccc(CO)c(F)c1 Cc1ccc(C(=O)NC2CN(C(c3ncsc3Br)=O)CC2C#N)c(C)c1 c1(C2(OC)CCCCCC2)ccc2oc(=O)n(C)c2c1.c12ocnc1CNCC2 N1(C(CSC)=O)CCN(C(c2c(C)cc(C)nc2O)=O)CC(C)(F)C1 c1(C(=O)NCCOC2CN(C(C(C)=C(CC)C)=O)C2)[nH]cc2c1CCCC2 c1(C(N(C(CNC(CC(C=C)C)=O)C)C)=O)cc(CC)nc(O)c1 C1(N(C(C2(C)CC2)CO)C(C2(C(=O)O)CC2)=O)CCOCC1 C(=O)(C(O)CCNC(c1ccncn1)=O)N(C(C)C)Cc1ccco1 Cc1ccc(CS(N2CCC(O)(c3ccccc3F)C2)(=O)=O)c(Cl)c1 N1(C(C2(C)CCSCC2)=O)CCC2(CCN(C(c3ccc(N)c(N)c3)=O)C2)C1 c1(NC(CC(=O)NC2CCN(CC)CC2C)=O)ccc2nc(C)cn2c1 c1(C(=O)NCCOCCNC(CC2(C)CC2(F)Cl)=O)ccc(=N)[nH]n1 Cc1cccn2nc(C(=O)NCC(C)CN(C)C(c3sccc3F)=O)cc12 C(=O)(CCCC(=C)C)NCCOCCOCCNC(CCC#C)=O C12(CNC(c3c(CC)noc3)=O)CCC1CCN2C(=O)C(C)=CC(C)(C)C c1(C(N2CC(NC(C(C)P(C)(C)=O)=O)CC2(C)C)=O)n[nH]c2c1COCC2 N1(C(C=Cc2cnc(C)s2)=O)CCCC(NC(=O)CC2(C#N)CCCCC2)CC1 Cc1nc(N2CC=CC(NC(C3Cc4ccncc4C3)=O)C2)c(F)c(C)n1 C1(CCC(=O)NCC2CCC(C(=O)NC3CC(CCF)C3)O2)CCC(O)CC1 c1(NC(C)=O)ccc(C(=O)NCCN(C(=O)C=Cc2ncc[nH]2)C(C)=O)cc1 N(C1c2ccccc2CC1NC(=O)C=CBr)C(=O)CCn1cccc1 CC(C)C(C(=O)OCc1nc(C2C(C)(C)C2(C)C)n[nH]1)C(C)NC(=O)C(F)(F)F N1(C(c2ccc(C#N)cn2)C(=O)NC(CC)(C)C)CC(=O)N(C)CC1C(=O)OC C#CC(CNC(=O)CNC(=O)CC1CCN(C)C1=O)CC(C)(C)C N1(C(c2c(C)onc2)=O)CCC(NC(=O)CCc2csc(=N)[nH]2)CC1C C12(NC(Cc3c(C)nc[nH]3)=O)CCCC1CN(C(c1cccc(O)c1F)=O)C2 N1(C(C23CC(NC(Cc4c(C)ccs4)=O)C(OC2)C3)=O)CC2CCN(C)CC2C1 c1(C(N(CCNC(=O)Cn2ccnn2)CC)=O)csc2cccc(F)c12 c1(C(=O)NC2C(C)CN(C(=O)C(c3ccc(F)cc3)=O)C2)nc(O)nc(O)c1F C1(NC(=O)CC2(CO)CC2)CCN(C(=O)CC2NC(=O)NC2=O)CC12CCC2 N1(C(c2c(C)nc(O)s2)=O)CC(C)(C)CC1CNC(=O)CC1CN2CCN1CC2 C1(C(N(c2ccccc2)CCOC)=O)CCN(C(c2ccnn2C(C)C)=O)C1 c1(CC(=O)NC(CNC(c2nc(C)c(C)s2)=O)C2CC2)cc(Cl)ccc1F C1(N(C(C2(NC(C)=O)CCC2)=O)C)CN(C(=O)C(C2CC(F)(F)C2)O)CC12CC2 Cc1nc2ccc(C(=O)NC3(CNC(=O)CCS(C)=O)CCC3)cc2nc1C c1(NC(C2CC(OC)C2)=O)ccc(NC(c2c[nH]c(=N)o2)=O)cc1C c1(CCC(=O)NCC(C(C)C)NC(C2CCC(O)C2)=O)nc2cccnc2[nH]1 C1(NC(c2n(C)nc3c2CCC3)=O)CCCC12CCN(C(c1ccsc1)=O)C2 C1(NC(c2cc(C)n(CCO)n2)=O)CCN(c2nnc(C(F)F)o2)C(C)C1 N1(C(c2c(Br)cn(C)n2)=O)CCC(NC(=O)C=CC2CCOC2)C12CC2 N1(C(CCN(C(c2cc(C)[nH]c2C)=O)CCO)=O)CCCC2(C1)N=N2 C(=O)(C(C)(C)C(F)F)NC(CC)CNC(C1(c2ccsc2)CC1)=O C1(NC(CN(C(C)C)C)=O)CN(C(=O)CC2(C)CC2(Cl)Cl)CC1(C)C N1(C(c2ccc(CNC(CSCCC)=O)nc2)=O)CCC2OCCC2C1 c1(CN2C(C)(CCC(N3CCC(F)CC3)=O)CCC2)ncc(C(F)(F)F)cc1Br CC(C(=O)N(CCC(C(C)(C)C)NC(C1(c2cccs2)CCC1)=O)C)C(F)(F)F c1(C(N(CCNC(c2csnc2OC)=O)CC)=O)cc(Cl)cc(F)c1F c1(OC)cccc(C(=O)NCC2(O)CC(C(=O)NCC3(OC)CCC(C)C3)C2)c1 c1(CC(=O)NCC2(C3N(C(CNC=O)=O)CCC3)CC2)sc(O)nc1O C1(C(=O)NCCOC(CC)CC)C(C)OCCN1C(=O)CC(CN(C)C)CC C(c1ccc2ncccc2c1)=CC(=O)NC1CC1C(=O)NC1(C)CCCCC1 c1(C(=O)NCc2ccccc2S)nnc2n1CC(C(F)(F)F)CC2 C(c1ccc(Cl)s1)=CC(=O)N(CCCN(C(C(C1CCC(C)CC1)CC)=O)C)C C1(N(C(=O)C(CO)c2ccccc2)Cc2ccccc2Cl)(CO)CCCCC1 C(=O)(CC(C(C)(C)C)NC(C1(C)N=C(C)SC1)=O)NC1CN(C2COC2)C1 C1(C(=O)NCCC2CN(C(C(CCC)CCC)=O)C2)CC2(C)CCCN2S1(=O)=O c1(CC(=O)NC2CC(NC(c3cc(CC)c(C)s3)=O)CC2O)cccc(C#N)c1 S(=O)(=O)(c1ccc(NCC2(CF)CCC2)cc1Cl)NCc1cccc(SC)c1C n1(CCCN(CC)CC)ccnc1CNC(=O)CCOC1CC1.C(CCC)SC c1(C(N2CCN(C(c3nnn4ccccc34)=O)C3CC23)=O)cc2oc(Cl)cc2[nH]1 CN1CCC(C(=O)NCC(C2CC2)NC(c2nn(C)cc2Cl)=O)CC1 C1(C(=O)NCC=CCC(=O)NC(c2onc(C)n2)C)CCC(C)(C)C1 C12(C(N(CC(CN(C(COCCN(C)C)=O)C)O)C)=O)CCCCC1C2 C(=O)(CCCCC(F)(F)F)NCC(C)CNC(=O)C(c1ccccc1)C1CC1 CC1CN(C(=O)CSc2ccc(Cl)cc2)CC1NC(=O)C(C)CO C1(C2CC2)(C(=O)NCC(c2ccco2)OC)CN(C(=O)CC2CCOC2C)C1 C1C(C)N=C2C=CC(Br)=C(S(=O)(=O)N1C)N2.C1(N)CCN(S(=O)(=O)CC)CC1.CS C=CC(O)C(=O)NCCOC1CN(C(c2ccc(CSC)s2)=O)C1 CCCC(=O)N(CC(C)O)C(C)=O.C(=O)(C(C)SC)N.C1CNCCCO1 C=CCCCC(C)N=c1nc2c(cnn2C)c(NCCN2CCCC(C)C2)[nH]1 O=S(=O)(c1[nH]c(=NCCCC2CCOC2)ccc1Br)NC1CCn2ccnc2C1 c1(CC(=O)NC(C2N(C(c3c(C)cnnc3)=O)CCC2)C)ccc(Cl)nc1C C12(C(N(C(C)COC)CC)=O)C(NC(=O)CC3CCCO3)C3CC1C2C3 C1(NC(CNCCCCC)=O)CCC(CCC(=O)Nc2c[nH]nc2OCC)CC1 c1(CNC(N(C(c2ccc(F)cc2)C)CC)=O)ccc2c(c1)CN(C)C2=O C1(C(=O)[N+](C(C2C(C(N(C(C=C)C3CC3)C)=O)C2)C)([O-])OCC)CC2(C1)CC21CC1 c1(CC)cc(NC(=O)C(O)C2CN(C(=O)CC(COC)COC)C2)cnc1C C(=O)(C(C)(C)CC(F)F)NCCCn1cc(C(C)N(c2cncc(Cl)c2)C)nn1 C(=O)(C(C)CC(=O)NC1CC(NC(C2CC3CCCC23)=O)C1)OC C1(CNC(C2CN(C)C2)=O)CCCN1C(=O)Cc1nnn(C(C)(C)C)n1 C(=O)(C(CCCC)NC(=O)C(F)C(C)(F)F)NCC(C#C)OC CCCCC(C(=O)NCC1CC2(CCC2O)C1)NC(C1CC2C=CC1O2)=O c1(C(=O)NCCNC(c2ccn(CC)n2)=O)ccnc(CC(C)C)c1 C1(CCC)CCC(C(C(=O)NC2CCOC2)N(C)Cc2cc[nH]n2)CC1 C#CCCN=C(NCc1nn(CC2CC2)cc1Br)NC(CCOC)c1ccco1 c1(CC2OCCN(C(=O)NCCOc3c(C)cccc3)C2)c(F)cc(I)cc1F N1(C(C(Cn2cccn2)NC(C(C)(C)C(F)F)=O)=O)CCC12CCC(O)CC2 C1(NC(C(C=C)CC)=O)CN(C(c2c[nH]nc2Cl)=O)C2(CCCC2)C1 c1(CN2C(=O)C(Cc3ccccc3)C3(CCC2)CC3)ccc(Cl)c(Cl)c1.CO c1(SCC)cc(C(N2CC(CNC(c3c(CC)csn3)=O)C2)=O)ccn1 c1(C2C(=O)O2)ccc(Br)s1.CCC(C)(C)OC(C)(C)C C1(C(=O)NCC2(C)N(C(c3c(C)nc(C)[nH]3)=O)CCC2)CCC(C)(C)CO1 C12(CNC(CC3(C)CC3)=O)CCCC1CCN2C(c1ccc(Br)o1)=O c1(C(=O)NC(C)(C)CCNC(C2CCOC(=O)CC2)=O)ccn2cncc2c1 c1(C(N2C(CNC(C=C(CC)C)=O)COC(C)(C)C2)=O)ccnc2c1ccn2C C(C1OB(O)c2ccccc21)NC(=O)CCc1ccncc1Br c1(NC(=O)Cc2cnccc2C(=O)O)ccc2c(c1)C(Br)(F)CC2 CC(F)(F)CCC(=O)NC1CN(C(C2CCCCCC2)=O)CC1CO O(NC(=O)C(CCSC)NC(C)=O)CCCC(=O)NCCC=CCCC C(=O)(CC(C)N(C(=O)CN(C)CCS)C)OC.CC(C)OC CCCC(CC(=O)NCc1noc(CC)n1)NC(c1cc(C(N)=O)c[nH]1)=O c1(NC(C(C)CO)c2nnnn2C2CCOCC2)cccc(-c2cnn(C)c2)c1 C1(O)(C(C(=O)OCC)(F)F)CCN(C(=O)C(C)N(C)Cc2ccccc2)CC1 N1(C(C(C2CC2)NC(c2cc(Cl)n[nH]2)=O)=O)CCC2(CCCOC2)C1 N1(C(C2CCCC(C)C2)=O)CCC2(CCN(C(=O)CC34COCC(C3)C4)C2)C1 C1(C(=O)NC(CNC(c2ccc(CC)[nH]2)=O)CO)CCN(C)C1=O C(CS(=O)CC(F)(F)F)NC(N1CCC(n2c(NC(C)=O)ccn2)C1)=O C(=O)(N=c1ccn(CCC(=O)OC)[nH]1)c1n(CC)ncc1Br C1(N(C(CC(CC)C)=O)CC2CC2(F)F)CCNCCC1C c1(C(=O)NCC(C)C)ccc(C(Cn2cc(CCCOC)nn2)OC)s1 c1(C(N(CCNC(C(CC)=CC)=O)CC2CC2)=O)ccc2cc[nH]c2n1 N1(C(C2(C)CC(C)(C)C2)=O)CC2(C1)CN(C(=O)C(C)(C)N1CCCCC1)C2 c1(C(=O)NC2CCCC(NC(CC(C=C)C)=O)C2)cc2c(s1)COCC2 C#Cc1cncc(C(N2CCN(C(C3SCC=C3C)=O)CC2CCO)=O)c1 N1(C(c2c(OC)ccc(F)c2)=O)CC2(CCCC2NC(c2cc(C)co2)=O)C1 C(=O)(C(C)(C)C(C)N(C)C)NCC1CC(N(C(C)=O)C)C1 c1(CC)nnc(C)cc1C(=O)NC(C)CCNC(c1ccc(OCOC)cc1)=O c1(OC)c(C)cc(C(=O)NCC2CCCC(CN(C(=O)C=CCO)CC)C2)cc1C C1(NC(C(C)OCCN(C)C)=O)CCC2(CC1)CN(C(C1CCCCCC1)=O)C2 C(=O)(C(CO)NC(C1CCCC1)=O)NCCN(C(=O)CC(C1CC1)C1CC1)C Cc1cc(=NCC2CCC3(C2)OCCO3)[nH]cc1S(=O)(=O)NCC1(C)CC1(Cl)Cl N1(C(COCC#C)=O)CC(CNC(=O)CCOCC(F)(F)C(F)F)C2CC12 N1(C(C(CCC)(C)O)=O)CCC(NC(C2CC3(CCCC3)CO2)=O)C(C)(C)C1 N1(C(=O)OC(C)(C)C)CCOCC1CC(=O)OCCCNC(=O)C(C)O Cc1cc(C(=O)NC(C)CCN(C(=O)CN2CCCNC2=O)C)sc1C N1(C(c2cc(C)nn2C(C)(C)C)=O)C(C)C2CC1C2NC(=O)CC1CN(C)C1 CC1CCC(CNC(=O)Cc2cc(C(F)(F)F)co2)N(C(=O)CCc2cnoc2)C1 C1(C(=O)NCCCCOC)(CF)CCN(C(=O)C(C)COC(C)=O)C1 C(C(CO)CC(C)C)NC(CCC1N(C(c2cc(C)nn2C)=O)CCCC1)=O C1(C(=O)NC2CC(CCNC(c3c(C)noc3)=O)C2)CCOCC1(C)C C1(c2n(C3C(C)(O)CCC3)nc(Cc3ccc(CO)cc3)n2)CCc2nn[nH]c2C1 C(=O)(C(F)(F)c1csc(C)c1)NC1CC(CNC(COCCC)=O)C1 CC1(O)CCCN(C(C2CN(C(=O)COC3CCOCC3)CCO2)=O)C1 C(=O)(C1Cc2ccccc21)N1CCCC(NC(C(CCSC)O)=O)(CO)C1 c1(OC)nc(C)ccc1-c1nccn1-c1cccc(C2NCCOC2)c1.C(C)C C1(NC(c2c(O)ccc(OC)c2)=O)COC2(C1)CN(C(C1(CF)CC1)=O)C2 N1(C(CC=CC(C)(C)C)=O)CC(C(=O)NCc2cocn2)C2(CC2)C1 c1(CCC(=O)NCC(CNC(CSCCC)=O)CO)cccc(O)n1 C=CC(C)(O)C(=O)NCC(C)NC(=O)C=C(C)Cl c1(C(=O)NCCCCN=[N+]=[N-])ccc(NC2CCc3ccccc32)c([N+](=O)[O-])c1 Cc1ncc(CCC(=O)NCC(C)(CO)NC(C2CC2C(C)C)=O)s1 N1(CCSCC(=O)NCCNC(=O)C(O)Cc2cnc[nH]2)Cc2ccccc2C1 Cc1cn2cc(NC(C3CC3NC(=O)Cc3nc4ncccn4n3)=O)ccc2n1 c1(C(=O)Nc2ccn3ncnc3c2)[nH]nc2ncc(-c3cccnc3CO)cc12 c1(NC(N2CCCC(C(C(=O)OC)O)C2)=O)nccc(C(N)=O)c1[N+](=O)[O-] N1(C(CCSC)=O)CCC(N(C(=O)CNC(=O)Cn2cncn2)CCO)C1 CCCCC(C)CCC(=O)N1CCC(N(C)C(c2ccc(Cl)cc2Cl)=O)C1 CC1CCOC(C(N2CCC(O)(CNC(=O)C(Cl)=CCl)C2)=O)C1 c1(C(=O)NCC2N(C(c3c(OC)ccs3)=O)CCCC2)cnc2ccc(Cl)cn12 c1(OCC)ccc(CC(N2CCC2CNC(c2cc(F)c[nH]2)=O)=O)cc1 C1(NC(C2CC3CCCCN3C2=O)=O)CCS(=O)(=O)C12CN(C(=O)C1CC1)C2 c1(CC(=O)NCC(CC=C)NC(=O)C(C)(CC)C(F)F)ccc(C)c(F)c1F C12(CC3(NC(C=Cc4c(C)ncs4)=O)CC3)CCC(CC1)N2C(=O)CCOC C1(SCC(=O)N(C(C)C)CCN(C(=O)C(C2CCOCC2)O)C)CCS(=O)(=O)C1 c1(C(N2CCC(OCCNC(=O)CCCC3CC3)C2)=O)ccn2cccc2c1 c1(C(N(C)C)=O)cccc(C(=O)NC2CN(C(c3cnc(N)cn3)=O)C3CC23)c1 N1(C(c2c(CSC)cccn2)=O)CCC(NC(=O)C=Cc2nc(C)cs2)C(C)C1 C1(NC(C(c2ccc(CC)s2)=O)=O)CSC12CN(C(C1(C#N)CCC1)=O)C2 O=S(=O)(c1cccc2c(Cl)nccc12)NC1CN(Cc2cnsn2)CC1F c1(OC)cccc(C(=O)NCC2CCCN(C(=O)C3=C(C)CCC3)CC2)c1F C1(n2cc(CCCC)nn2)CC2CCC1(NC(C1CCSC1)=O)C2 N1(C(C2(CC)CCCO2)=O)CCC(C(=O)Nc2cccnc2)C(C)C1 c1(C(c2nnnn2C2CCOC2)NC(C(C)(C)OC(C)C)=O)cccc(Br)n1 N1(C(CCC=C(C)C)=O)CCC(C)(C)C(C(=O)N(C)CCOC2CC2)C1 N1(C(C(C)OCCC(C)C)=O)CC2CC1C2NC(c1nccn1C)=O c1(C(=O)OC)c(C)cc(NC(c2ccc(F)c(-n3cc(CO)nn3)c2)=O)nc1C C1(NC(C(CCOC)C)=O)CC(C)CN(C(=O)Cc2ccsc2Cl)C1 N1(C(COC)OC)CCC(CC(N2CCSCC2)=O)C1 c12ncnc(c1Br)N2SC.c1(C)ncc(Br)cc1F.C1(O)CNC1 c1(C(=O)NC2CC(C(C)N)C2)cc(-n2cncn2)ccc1Cl C1(OC)CC2CC(NC(=O)C(=O)NCC3(Oc4ccc(Cl)cc4)CCCC3)CC12 N1(C(c2c(C)nn(CCO)c2)=O)CCC(C2CC2NC(c2nnsc2C)=O)CC1 C1(NC(c2n(C)c(O)nc2)=O)CC2CN(C(C3(C(F)F)CCCO3)=O)CC2C1 c1(NC(C23C(CN(C(CCOC)=O)C2)C3)=O)ccc(Br)c(Cl)c1 C12(C(=O)NC3CCN(CCC)C3)COCC1CN(C(c1ccc(C#N)cc1)=O)C2 c1(C(=O)NCCCCN(C(=O)CCSCC(N)=O)C)ccc(C(F)F)cn1 c1(C(N2CC(C(C(=O)N(CC(C)O)CCF)O)C2)=O)sccc1F N1(C(C(C)(C)OC)=O)CCCC(F)(CNC(c2cn(C(C)C)cc2C)=O)C1 CC1CCC(C(=O)NC2CC3(CCC3)C2O)N(C(c2cocn2)=O)C1 c1(C(=O)NCC2(CNC(Cn3c(C)cnc3)=O)CC2)ccc2c(c1)CCCS2 C1(OC)CN(C(c2cnn[nH]2)=O)CCC1NC(c1cccc(OC(C)C)c1F)=O C(=O)(CCCCCCN=[N+]=[N-])NC(CCN(C(C1CC2(ON=C(C)C2)C1)=O)C)C Cc1cc(C(F)(F)F)sc1C(=O)N(CCNC(=O)C(C1CCCCC1)O)C(C)C c1(N2CCC(N(C(=O)C3=C(C)CCCC3)CC#C)CC2)cnc(C#N)c(C#N)n1 N1(C(c2cccc(OCC)c2)=O)CCC(NC(C2CC(C#N)C2)=O)CC1C c1(C(=O)NC(C2(O)CN(C(=O)CC3CCNC(=O)C3)C2)C)cc2c(s1)CCOC2 c1(C(N2C(C(=O)NCCC3CCOC3)COCC2)=O)cccc(F)c1F c1(C(=O)OC)ccc(F)c(C(N2CC=CC(NC(C34CC(C)C3C4)=O)C2)=O)c1 Cc1cc(C(=O)NCC(C)N(C)C(C2CC(CN(C)C)C2)=O)c(C)cc1Cl C1(NC(c2c(OC)cc(C)s2)=O)CCCCN(C(=O)C(C)(O)c2ccccn2)C1 C1(C(N2CCC(C)CC2C)=O)CC2C=CC1N(C(=O)Cc1ccnc(O)c1)C2 C(=O)(C(C#N)C(C)(C)C)N1CC(CC(=O)NC2CC(CSC)C2)C(C)C1 c1(CC(N2CC3C(C(N4CCC5(CC5)C4)=O)C3C2)=O)n[nH]c2ccccc12 C(=O)(CCC(=O)N1CCC(C(=O)NCC2=C(C)CCC2)C1)NC CCCC(C)(O)CC(=O)N(CCCNC(c1cc(Cl)c(Cl)n1C)=O)C1CC1 C1(CC(=O)NCC2N(C(C(C)CF)=O)CCN(C)C2)Cc2ccccc2N1 c1(N2C(CC(C)NC(C3(c4cccs4)CC3)=O)CCC2)ccc(C#N)nc1 Cc1ccc(-c2nc(CCC(C)C)nn2C)cc1Br c1(CC(N2C(C(=O)NCC(CC)N(C)C)CC2)=O)cc(C)on1 c1(C(=O)OC)ncnc(C)c1N1CCN(C(C2CN3CCC2CC3)=O)CC1 C1(CNC(C2N(C(C(C(C)O)N(C)C)=O)CSC2)=O)COCC(=O)N1C N1(C(C2(OC)CC2)=O)CCC(O)(CN(C)C(c2cccc(SC)c2)=O)C1 c1(C(=O)NCC2C(NC(=O)CCSc3ccccc3Cl)C2)ncc2ccccn12 CCC(O)C(C)(C)C(=O)N(CCCNC(c1noc2ncccc12)=O)CC c1(OC(C(N2C(CC#C)CCC2)=O)C)cc(C)ccc1Cl c1(NC(C2CC(=C)CN2Cc2ccc(N(C)C)cc2)=O)c(C)cccc1Br c1(C(N2CCC(N(C(=O)CCCC(C)=O)CC)C2)=O)cc(=O)c2ccccc2o1 C1(C)(CN(CC(=O)NC2CC(F)(F)C2)C)CCCN1C(=O)CCS(C)=O N1(C(C2C(NC(=O)CC3(O)CCC3)CC=CC2)=O)C(CO)CCC12CCC2 C1(C(N(C)CC2CCN(C(c3cc(O)ccc3F)=O)C2)=O)CCC12CCOCC2 Cc1noc(C)c1C=CC(=O)NC1CC(C)N(C(c2cnc(C(C)(C)C)s2)=O)C1 c1(C(=O)OC)ccc(C(=O)N(CCCNC(C2CC2[N+](=O)[O-])=O)C(C)C)cn1 C1(CNC(c2c(OC)cccn2)=O)CN(C)CCN1C(=O)C(C)NS(C)(=O)=O N1(C(C(C)Oc2ccc(C#N)cc2)=O)CC(NC(=O)CC2(C)CC2)CC1(C)C N1(C(C(CC)c2cccnc2)=O)CCCC(N(C)C(c2ccc(N)cn2)=O)C1 c1(C(N2CCN(C(c3occ(C)c3)=O)C(CO)C2)=O)cc2c(Cl)cccc2[nH]1 CC1(C)COCCN(C(C2COCCC2NC(=O)CC2CCSC2)=O)C1 CC1CC(CC(=O)NCCNC(=O)C(C)(C)C)CN1C(C1CC2CCC2C1)=O CCC(CC(F)F)C(=O)NCC(C1CC1)NC(c1cnc2[nH]ncc2c1)=O C1(O)(CCNC(C(C)N(C(C)=O)C)=O)CCN(C(=O)C(F)n2ccnc2)CC1 Cc1nccc(Cl)c1C(=O)N(C1CCN(C(C2CCOCC2)=O)CC1)CC1CC1 N#Cc1cc(C(=O)NCC23CC2CN(C(=O)C2=C(Cl)CC2)C3)co1 CC1=C(C(=O)NCC2(F)CN(C(=O)Cc3scnc3C)C2)C(C)(C)CCC1 Cc1cc(C)c(C(=O)NC(C)(C)C(C)NC(c2cncn(C)c2=O)=O)cc1N Cc1cc(NC(=O)NC(C)(C)C)ccc1NC(=O)CC1CCCCC1 Cc1c(C(=O)N(C2CC(NC(C)C)C2(C)C)C)ccc2ccccc12 N1(C(C(C)NC(c2ccc(C)cc2)=O)=O)CC2CC(C1)C2NC(=O)C(F)C(C)C c1(C(N2CC(NC(=O)C=CC3CCC3)CC(C)C2)=O)n[nH]c2ccc(F)cc12 N1(C(C(c2ccc(C)s2)C)=O)CCCCCC1CNC(c1ccc(F)cc1N)=O c1(CCCC)ccc(NC(Cc2cccc(C)c2)C(C)C)c(Br)c1N C1(CNC(C2CC(OC)C2)=O)(NC(C2(C)CC2(F)Cl)=O)CCCCC1C CC(C(=O)NCC1(O)CCN(C(C23CCC(F)(CO2)C3)=O)CC1)C(C)(C)C c1(CN2C(NC(C3CN(CCCO)CCO3)=O)CSCC2)cc(I)ccc1Br c1(C(N(CC(C)(C)CCO)CC)=O)cccc2c1CCCC2=O C(CN=c1[nH]c(C2CCCC2)nc(=N)[nH]1)N(C(=O)COCc1ccc(F)cc1)C c1(C(=O)NC2(CCCNC(=O)CC3CCCCO3)CC2)noc2c1COCC2 C12(C(=O)NCC#CC(=O)NCC(F)(F)F)CC1CNC2=O N1(C(c2nc(CNC(c3cc(C#N)[nH]c3)=O)oc2)=O)CC2(CCCC2)C1 C1(C(=O)NC2CN(C(c3c(C)ncc(C)c3)=O)CC(C)C2)CCn2nnnc2C1 Cc1cc(C(=O)NC2COCCN(C(=O)CN3CCCCCC3)C2)nc(Cl)c1 C1(C(=O)NC(C(=O)NCC)C)CCC(C)(C)N(C)C(=O)CC1CSC N1(C(C=Cc2c(C)nccc2)=O)CC2CCN(C(=O)CC(C)P(C)(C)=O)C2C1 C(=O)(C(CC1CCCC1)NC(=O)CCCOC(C)(C)C)N(CCC(N)=O)C C=CCCCC(=O)NCC(c1ccc(F)cc1)NC(=O)COCC(C)OC C1(CNC(C2C(COC)C2)=O)CN(C(c2c(F)cncc2Cl)=O)CC2(CCC2)O1 N1(C(c2ccc(CNC(C#CC(C)(C)C)=O)cc2)=O)CC(C2CCCC2)C1 c1(OC)ccc(C#N)cc1CNC1(c2ccccc2C#N)CC1 c1(NC(C(=O)NC(=O)NCCN(C2CC2)C2CC2)=O)ccccc1[N+](=O)[O-] C(=O)(CCC(C)(C)C#N)N1CCCC(NC(c2c(CC)nns2)=O)(COC)C1 c1(NC(C(N2C3CN(C(C4CC(OC)C4)=O)C(C3)C2)=O)=O)ccc(C#N)c(Cl)c1 c1(C(N2CCC(N(C(c3c(C)c(Br)ccc3)=O)C)C2)=O)ccnc2ccnn12 C1(NC(c2cc3ccccc3[nH]2)=O)CC2CCC1CN2C(=O)CCC(F)(F)F C1C(C)(C)CC(=O)OCC2(CC2)C(=O)N1.C1(CC)CCCCC1C(=O)OC CCCCC(CNC(=O)C)N.c1(C2C(NC(c3ccc(CO)s3)=O)C2)cnn(C)c1 C1(S(C)(=O)=O)(CN2CCN(C(COC)(C)C)CC2)CC(O)(C(=O)O)C1 N1(C(CC(CCC)CCC)=O)CCC2CN(C(=O)C3CC3)CCC2C1 C1(C(C)NC(c2cc(N)ccn2)=O)CN(C(=O)C(C)(C)c2ccccn2)CCO1 CC1(C(N2CCC(CNC(C3(CC4CC4)CC3)=O)CC2)=O)CC(F)(F)C1 c1(C(=O)NCC2CN(C(c3c(C)onc3)=O)C(C)C2)ccc(=O)n(C(C)C)c1 C1(C(=O)NCCOCC(C)NC(CC2(COC)CCCC2)=O)CCC(C)(C)CC1 c1(C(N(C(c2ccccc2)C(C)=O)C)C)cn(C(C)C(=O)OC)nn1 Cc1cc(Br)cc(Cl)c1CN1CCCC1C(=O)NCC(C)C c1(N(C)CCNC2CN(C)CCO2)nc(=NCC2CCOCC2)[nH]c2c1COC2 N1(C(N2CCc3ccccc3C2)=O)CCCC2CN(c3cccnc3)CCC12 N1(C(c2c(OC)ccnc2Cl)=O)CCCc2c(OC)ccc(C)c21 c1(C(N2CC(O)(CNC(C(CCC)(C)C)=O)C2)=O)cc2ccccc2c(=O)o1 C(=O)(C1=CC2CCCCC12)NCC(CCOC)NC(c1cc2sccc2[nH]1)=O N1(C(c2nn(CC)c(O)c2)=O)CCC(C2CCN(C(=O)C=CC(C)C)CC2)C1 C1(NC(CC(C)C)=O)COC2CN(C(=O)CCF)CC12 C=CC1CCN(C(C2CCCN(C(C3CCC3C#N)=O)C2)=O)C1 C(C(COC)C(=O)NCCCCCCNC(C1CCOC(C(C)C)C1)=O)OC c1(CN2CC3CCN(S(=O)(=O)CCCCl)C3C2)cccc2nscc12 C1(NC(C2(C)CC(NC(CCn3ccc(C)n3)=O)C2)=O)CC2(CC(=O)C2)C1 C1(C(C(=O)N(C(C)C2CC2)C)F)CCN(C(=O)C(C2CCOCC2)F)CC1 Fc1cccc(C(c2nnnn2CC)NC2(C(F)F)CC(C(F)F)C2)c1.C1CCC1 c1(CNC(N2CCC(C)(OC)CC2)=O)nc2c(s1)CC(C(C)(C)C)CC2 c1(C(=O)NC2C(CCOC)C2)ccc(CNC(=O)CN2CCC(C)CC2)nc1 Nc1nc2c(cc1C(=O)NCCC1CC(NC(C3CCS3(=O)=O)=O)C1)CCCC2 C1(CCC)CN(C(C2CC23CC(OC)C3)=O)CCN1C(=O)C=C(Cl)Cl CC(CC(=O)NCCCCC1CN(C(C2CC3(CCCO3)C2)=O)C1)CC(C)(C)C C(CC#CC)(C(=O)NC(CC)CC(F)(F)F)NC(CCC=CCC=C)=O c1(C(N2CC3CC3(CO)C2)=O)cnc2c(-c3ccnnc3)cccc2c1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCN(C(c2c(C)n(C)cc2)=O)CC1 C1(NC(C(C)=C2CC2)=O)CCCC1CNC(c1csc(O)n1)=O c1(CN2CC3N(C(C4(OC)CC4)=O)C3C2)nccc2ccccc12 S(=O)(=O)(c1c[nH]c2cccc(F)c12)N(C(C)CCO)CC(C)(C)C c1(C(C(=O)NCCOC)N(C(C(=O)OCC)C)C)nn(C)cc1C C(C(CNC(=O)CC12CC(CO)(C1)C2)CO)NC(CNC(=O)OC)=O c1(C(=O)NCCCS)ccnc(C2CC2)c1.C(CC(=O)N(C)CC)OCCN(C)C c1(C(=O)NCCCCNC(c2cc(O)nc(Cl)c2)=O)cc(F)c(CO)c(F)c1 C1(CNC(C(C)OCC#C)=O)CCCCN1C(=O)C(=O)N(C(C)COC)C N1(C(c2n(C)ncc2Cl)=O)Cc2ccccc2C(NC(=O)CC(C)(C)C#N)C1 c1(OC)ccc(F)c(C(=O)NCCOCCCNC(C2(C)CC2)=O)c1N.C1(SS)CC1 C1(NC(CC(=O)NC)=O)CN(CC)CCC1C.c12cc(nc(C(F)(F)F)n1)N2 C1(CNC(C2CCCN(C(c3cc(C)ncn3)=O)C2)=O)CCC2(CCC2)O1 c1(CC)cc(Br)cc(S(=O)(=O)NNC(=O)c2ccn(C)c2)c1 CCC(CNC(C1CC(NC(C2CCCC2)=O)C1)=O)CC(C)C c1(SC)ncc(C(=O)N(C(C)CNC(C2(C(C)C)COC2)=O)C)n1C C(=O)(NN1CCCc2ccccc21)c1nc(OC)c(Cl)cc1 c1(OC)cccc(CO)c1.c1(C2N3CCC(F)(C3)NC2=O)cccc(F)c1 c1(C(=O)NC2C(CC)CN(C(=O)CCc3cccnc3F)C2)n[nH]cc1[N+](=O)[O-] C(C)(CCCCCO)NC(CC(CNC(C1(CC)CCCO1)=O)C)=O c1(C(=O)NCCCN2CCN(C(CCS(C)=O)=O)CC2)cnc(C(F)(F)F)c(F)c1 N1(C(COCCCCC)=O)CCC(CN(C(=O)CSCC(F)F)C)CC1 N1(C(COCC)=O)CC2OCCN(C(c3cncc(COC)c3)=O)C2C1 c1(CCC(=O)NCCN(CC)SCCO)ccc(OC2CCCC2)cc1.C1CS1 c1(C(N2CC(C(C)NC(C=CCCC)=O)C2)=O)nnsc1-c1ccccc1 N1(C(C(CC)=CC)=O)CC2CC(C1)CN(C(=O)CCC1CCCO1)C2 C1(CC#N)CCC(C(=O)NC2CCCC(C(=O)NC3CCCCC3CO)C2)CC1 c1(CCN(C)C(=O)NC2C(COC)(CC)C2)ncsc1OC.C1(O)CC(F)(F)C1 N1(c2n(CCSCC(C)C)c(-c3ccccn3)nn2)CCOC2(CNC(=O)N2)C1 C1(CC(=O)NCC2CC3CC3C2)C2CCCC2N1C(=O)C=CC1CCCC1 n1(-c2c(C(=O)NCC(CNC(CC=C)=O)OC)nccc2)ncc2ccccc12 c1(C(=O)OC)cc(NC(=O)Cn2cc(CSC)nn2)c(C)o1 CC1(C)C2CCC(C(N3CC4CCC3CC4NC(C3CCCCO3)=O)=O)C1C2 Cc1nc2ccc(C(=O)NC3CC(O)CN(C(=O)Cc4cnns4)C3)cn2n1 c1(CC(=O)N(C2CCN(C(=O)C3=COCC3)CC2)CC)cc(C)cc(F)c1 c1(CN2CCC(NC(c3ncc(Cl)cc3Br)=O)CC2)cc2cc[nH]c2cn1 C1(NC(C(C)OC2CCCC2)=O)CCCCCC1NC(=O)CC1COCCN1C Cc1c(C(=O)NCC2(NC(=O)Cc3cnns3)CCC2)cncc1Br CC1C(C(=O)N(C2CCN(C(c3cc(O)ncn3)=O)C2)C)OC2CCCCC12 C(=O)(CCC1=CCCCC1)N1CCCN(C)CC1CO NS(=O)(=O)c1ccc(CN2CC3CC2CN3C(C2CCCCO2)=O)cc1 C1(C2CCN(C(=O)C(c3ccnn3C)C)C2)(NC(C2CC(SC)C2)=O)CC1 N1(C(c2n(CC)c(O)nc2)=O)CCN(C(c2csc(C#N)c2)=O)CC(CO)C1 c1(OC)c(C(=O)NCC(C(C)(C)C)NC(C2C(Cl)(Cl)C23CC3)=O)csc1Cl C(CN=C(NCc1ccn(-c2cccc(Cl)c2)n1)N1CC(F)(F)C(F)(F)C1)OC C(C(CO)(CO)NC(C1CCCCN1C(C)C)=O)N(C(C(COC)C)=O)C C1(=CC(=O)NC2CCN(C(C(CC)F)=O)C(C)C2)CCOc2ccccc21 N1(C(C(C)(CSC)NC(C=CC(CC)C)=O)=O)CCC(CO)C(O)C1 C=C(C)C(C)(C)C(=O)NC1CCCN(C(c2cnn(C(C)(C)C)c2Cl)=O)C1 C1(C(N2C(C(N(C(CC)(C)C)CC(C)C)=O)CC2)=O)CCNC1=O C1(C(=O)NCC2(OC)CCC2)(C(F)F)CC(NC(=O)C(C)O)C1 C(C(C)CC(=O)NCCCC(C)(F)F)n1cc(CC(=O)OC)nn1 C(=O)(C(C(C)CC)NC(=O)CN1CCCCC1)N(CCCCCC=C)C Cc1cc(C(N2CCCCC2C2CCCN(S(C)(=O)=O)C2)=O)oc1C CC1=NC(C)(CNC(C2CCC(CNC(c3nccnc3N)=O)O2)=O)CS1 C(C(C)C(C)C(=O)N1CCCC1CNC(=O)C(C1CC1)C1CC1)OC CC(C)CC(O)CC(=O)N(CCCCC(=O)NC1C(C)CCC1C)C c1(C(=O)NCCC(C)NC(CCOC(CC(C)C)C)=O)cc(Cl)c([N+](=O)[O-])[nH]1 N1(C(c2ccc(CN(C)C)[nH]2)=O)CCCN(C(=O)CC2SC(=N)NC2=O)CC1 C12(C(=O)NC3C4CN(C(c5cc[nH]c5)=O)CC34)CCCC(C1)C(=O)NC2 c1(C(=O)NCC(C2CCOC2)NC(C(C)(C)c2cscc2Cl)=O)csc(C#N)c1 c1(C(N(CC(CC)NC(=O)C(n2cc(Cl)cn2)C)C)=O)ccc2sccc2c1 N1(C(c2n(CCN(C)C)ncc2)=O)CCC(N(CCO)C(C2CCCS2)=O)CC1 N1(C(c2ccc(C)cc2F)=O)CCC(NC(=O)C(C)CO)CC(C)(C)C1 C1(CNC(C2C(C(C)(F)F)C2)=O)CCCN(C(=O)CN2CC3CCC2C3)C1 C1(CC(=O)NCC(=C)Cl)CCCCN1C(=O)Cc1cnns1 N1(C(c2c(CC)ccs2)=O)CCN(C(C2C3CC3C3CC23)=O)CC1C Cc1ncccc1C(=O)NCCCCN(C(=O)C(F)CC1CCCC1)C CC(CC(=O)NC12CC(C(=O)N(C)OCc3ccccc3)(C1)C2)C1CCCO1 N1(C(c2c(C)cn(C)c2)=O)CCN(C)CC1C(=O)NCCc1ncoc1C N1(C(Cn2cccc(C)c2=O)=O)CC2CCCC2(NC(=O)CC(F)(F)F)C1 C(=O)(C1CCCc2ccnn21)NC(CC)CNC(c1cc(F)c(C#N)c(F)c1)=O c1(C(N(C2CCCN(C(=O)CC3C=CCCC3)C2)C)=O)cc(O)c2ccoc2c1 N1(C(CC2(COC)CCCC2)=O)CCCCC(NC(c2ccc(Cl)cc2)=O)C1 O=S(=O)(CC1CCOC(=O)CC1)N1CC2(CC2CO)C1 CC1(C)CSCCN1C(=O)C(C#N)OC1CCCC1 C1(CC)CCCN(CC(=O)NC2(C)CN(C(C3CC3C(C)(C)C)=O)C2)C1 C1(C(=O)NCCNC(c2nocc2Br)=O)CN2CC3CC2(CO1)C3 C(=O)(C1=C(C#N)CCC1)N1CC(CC)N(C(c2n[nH]c(C)c2C)=O)CC1 C(C(=O)Nc1ccn(CC(C)C)n1)(C(C(C)C)OC)N(C(CC)C)C.C1(C)CC1 N(S(=O)(=O)N1CCCc2ccccc21)c1c(C)ccc(F)c1 CC1CN(C(=O)CCOC2CC2)CCN1CC1CC1.C1(O)CCCO1 c1(N2CCC(C)C2)nc(N2CC3CN(C(=O)C4CC4)CC3C2)nc2ccsc12 CCCCCCn1nnnc1C(C1(Cl)CC1(F)F)NCCCSCCC(=O)C(C)C.N N1(C(C2C(OC)C2)=O)CCCCC1CCNC(c1cocc1C(N)=O)=O Cc1cncc(C=CC(=O)NCC2CCN2C(c2cc(Cl)c(Br)cn2)=O)c1 CCCCC(C)(F)C(=O)NC1CN(C(c2ccc(C#N)cn2)=O)CC1SC c1(C(=O)NCC(C2CCC2)NC(=O)CN2CC3CC3C2)cc2n(n1)CCNC2=O Cc1ccc(C(=O)NC(C2CCCC2)CNC(=O)CN(CC(C)(C)C)C)nn1 C1(C(=O)NCCCC(C)NC(c2cc(Cl)c[nH]2)=O)CCCC2CC12 Cc1cc(C(=O)NCc2ccoc2C(=O)NC(C)CC2CCCCC2)cc(C)c1 CC1CN(C(=O)C(C2CC=CCC2)NC(=O)CCCC2CC2C)Cc2nncn21 N1(C(CC(=O)OC)=O)CCN(C(=O)C=C2CCC2)CC1c1nccn1C C#Cc1ccc(C(N2CCC(OCCNC(=O)CC3CCC(C)CC3)C2)=O)o1 CC(C)CC(C)(CNC(=O)CCF)NC(c1ccc(Cl)cc1C(F)F)=O CC(CC1CC1)C(=O)NCCCOCCNC(=O)Cc1sccc1Cl C1(C(C)NC(C=CC(=O)NC2CN(C(=O)CN(C)C3CC3)C2)=O)CCN(CC)C1 N1(CC(=O)N(C2CCC(NC(=O)CNc3nccs3)C2)C)C(=O)NC(C)(C)C1=O c1(C(=O)NC2CC(C)N(C(=O)C3=CCCCC3)C2)cc(F)cc(F)c1F c1(CNC2CC(C(=O)NCC3COC3)C2)ccc(Br)cc1I N1(C(CCCCC=CCCC)=O)CC(C)(C)OCC1CNC(=O)C=CC1CC1 C12(CNC(C3CC(CC)OCC3)=O)CN(C(C3CC=CCC3)=O)CC(F)(C1)C2 c1(C(N2CCC(C(=O)OC)(OC)C2)C(=O)NC)ccc(-n2ccnc2)cc1 C1(C(=O)NCC2(CN(C)C(C3CCS(=O)(=O)CC3)=O)CC2)(OC)CCC12CCC2 C(=O)(C(C)(C)C(C)C)NC1CCC(N(C(c2cn(CC(C)C)nc2)=O)C)C1 c1(C(C)C)ncc(C(=O)NC2(C)CN(C(=O)C(O)CCn3cncn3)C2)n1C c1(CSCC(=O)NCC(CC)NC(C2CC(=O)N(C(C)C)C2)=O)ccccc1O c1(CC(=O)NC2CN(C(C3CC(O)C3)=O)CC3CC23)c[nH]c2ccccc2c1=O CC1CCCn2cc(C(=O)NC34CC(CNC(=O)C(C)C5CCCC5)(C3)C4)nc21 c1(OC)ccc(F)c(C(=O)NC(C)(CNC(c2cnc(N)cn2)=O)CC(C)C)n1 N1(C(CCC)C)CC(C(=O)NCC2CC2NC(=O)CSCCN(C)C)CC1=O Nc1cc(Cl)nc(Cl)c1C(=O)NCCN1CCN(C(C2CC(F)(F)CS2)=O)CC1 C1(CC=O)COCCO1.c1(C2CNC(=O)C2)ccccc1.N1(C(C)=O)CCC1CC CCCCCCCC(=O)N1CC2CC(C(=O)Nc3cnc4c(c3)CCC4)C(C2)C1 c1(CC)nc(C(=O)NCC(C)NC(=O)CC2CC2(Cl)Cl)c(N)s1 N1(C(c2c(CCC)nns2)=O)CC2C(CN(C(=O)C(C)C3CCC3)C)C2C1 C1(CCNC(CS(=O)(=O)NC)=O)C(C)CCCN1C(c1cccc(SC)c1)=O N1(C(C(c2cccc(C)c2)C)=O)CCCCC(NC(c2ccc(F)c(N)c2)=O)C1 c1(C(N2CC(C)CC2C)C(=O)NCCC)cncc(C)c1 CS(=O)C1(CO)CCN(C(c2sccc2OC)C(=O)NCc2ccco2)CC1 n1(CC=C)cc(C(=O)N(CC(C)N(C(=O)C(C)NC(C)=O)C)C)nn1 c1(C(=O)NCC2(NC(C3C(CC)C3)=O)CC2)cccc(N2CCCC2=O)c1 N1(C(Cc2ncn(C)c2)=O)CCC2CCN(C(=O)CS(N)(=O)=O)CC12 c1(C(=O)NC23CC(CNC(C=COCC)=O)(C2)C3)cnccc1C Cc1ccc(=O)n(CC(=O)NC2(C)CCCN(C(C3CN(C)C(=O)N3)=O)C2)n1 C123CCCC(CN1C2)C3.CCC1C(=O)N1.c1(SCc2ccccc2)nnsc1C C1(CC(=O)NC2CC3CC(C2)N(C(=O)C2=C(Cl)CC2)C3)CCC2(CC1)OCCO2 Cc1cccc(-c2c[nH]cc2C(=O)NC2COCC2CNC(=O)C(Cl)=CCl)c1 C1(C(N2C(C(N3C(C)(C(N(C)C)=O)CC3)=O)CC2)=O)COCC1(C)C N1(C(C=Cc2occ(C)n2)=O)CC2(CC(NC(c3cn(C)nc3C)=O)CO2)C1 C1(C(=O)NC(C(CO)NC(CSc2cccc(OC)c2)=O)C)CN2CCC1CC2 CC1(C)CCCCCC1NC(C1(CNC(=O)Cn2cnnn2)CC1)=O c1(OC)ccc(C(=O)NC(C(=O)NC2(CCCF)CC2)C2CCOC2)s1 N1(C(C(c2ccc(C)cc2)=O)=O)C2CCC1(CNC(=O)CCC1CC1(F)F)CC2 C1(CNC(CN2CCC(OC)C2)=O)CN(C(C2(CO)CCCO2)=O)CCCO1 C(C(O)(CNC(=O)CC1C2CN(C(=O)Cc3cncnc3O)CC12)CO)OC N1(C(CC(C)N(C(c2c(CC)csc2)=O)C)=O)CCCC(F)(CO)C1 N1(C(c2cccnc2)=O)CCC2OCCN(C(c3ccc(Cl)o3)=O)C2C1 c1(SC)nc(C)cc(=NC(C(C)NC(c2ccncc2)=O)C(C)C)[nH]1 CC1CC2CN(C(C3(C)CCCN3C(=O)CCc3ccccc3)=O)CCN2C1 CCCC(C)CC(=O)NC1CC2CC1N(C(c1cc(C(F)F)n(C)n1)=O)C2 C12(NC(c3cn(CCC)nc3)=O)CCCN(c3ccc(C#N)nn3)CC1C2 CC1=CCC(C(=O)NC2CC(NC(C3CCCN3c3cnccn3)=O)C2)CC1 C(=O)(CCCCCNC(N)=O)NC(CC)CN(C)C(c1oc(CO)nc1C)=O C1(NC(c2nocc2Br)=O)CCC2(CCCN2C(=O)CC2=CCCC2)CC1 N1(C(=O)OCC)CCN(C(=O)Nc2cc(C(C)C)n(C(F)F)n2)CC1C C1(NC(c2c(F)cccc2Cl)=O)CC2CC(C1)N(Cc1noc(C3CC3)n1)C2 N1(C(CC=CCC)=O)CC(C(=O)N(C)Cc2ocnc2C)CCC1(C)C Cc1cc(C)c(C(=O)NCCN(C(=O)C(c2ccccc2F)C)C(C)C)c(O)c1 N1(c2nc(COC)nc(C)c2)CC2(C)CN(C(C3CC3(C)C(C)C)=O)CC2(C)C1 N=c1nc(CCC(N2CC(O)(C(F)C(=O)NCc3ccncn3)C2)=O)[nH][nH]1 Cc1cc(C(=O)NCC(C2CCCN2C(C2NC(=O)CC2C)=O)(C)C)nc(O)n1 C(=O)(C(C(=O)N(C)CCC)OC)OCC.C1CCCCCNC(=O)CC2(CCC2)O1 c1(C(=O)NCC(C(C)C)NC(CCC)=O)ccc(OC(F)F)nc1Cl CCCCCCC(CC)C(=O)N1CCC2(CCN(C(C3(C)CCSCC3)=O)C2)C1 c1(C(N2CC(C)CC2C(C)C)C(=O)NCCOC)c(Cl)nc2sccn12 C1(CN(C)C(C2CCC(C(N)=O)O2)=O)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1 C12(C(=O)NC3CCN(C(C4CN=CCC4)=O)C3)CC3CC1C2C3(F)F C1(CNC(CCSCC)=O)(NC(=O)C(c2cccc(O)c2)C)CC2CCC1CC2 N1(C(Cc2cc(C)c(C(=O)O)o2)=O)CCN(Cc2cc(Cl)cc(Cl)c2)C(C)C1 C(C(CC(=O)N(C(C)CC(F)(F)F)C)NC(=O)C(C)(F)c1ccon1)OC c1(CC(N2C3C(C)(CCC3)C2)=O)c[nH]c2c(F)cccc12 CC1(C)CCN(C(=O)Cc2cncs2)C(C(=O)NC2CCSCC2)C1 N1(C(CCOCCN(C(c2ccc(C)cn2)=O)C)=O)Cc2c[nH]nc2C1 C(=O)(C(F)(CNC(c1ccn2cncc2c1)=O)C(C)C)N1C(COC)COCC1 c1(C(=O)NCC2(NC(C3CCC(F)C3)=O)CCOCC2)ccc(Cl)cc1Br c1(C(=O)NC2(CNC(C(COC)O)=O)CCOC2)cccc2nc(C)cnc12 c1(OC(C)C)cc(OC)cc(C(O)CNC2CC3CCC2(N)C3)c1 C12(COC)CCC1CCN2C(=O)CCNC(=O)OC(C)(C)C C1(CNC(c2c(C)ccs2)=O)CN(C(=O)CSCCN(C)C)CC(C)(C)C1 CCCCS(=O)(=O)NC(C)C(=O)NC1CCCCC1NC(C1CC(C(F)F)C1)=O C1(NC(C(=O)NCCOCCCC)=O)CCCN(C(c2cscc2F)=O)CC1 C1(C(=O)NCC2(C(N)=O)CN(C(=O)C3=NOCC3)C2)CN2CCC1CC2 C=Cc1ccc(C(=O)NC2CCN(C(c3[nH]cnc3C)=O)C(C)C2)cc1 CC1CC(N(C(=O)CNC(=O)CNC(=O)C(C)(C)n2cccn2)C)CC(C)C1 C1(C(N(CCN(C)C(c2c[nH]c(=O)cn2)=O)C)=O)CC(c2ccccc2)=NO1 c1(C(=O)NCCC(C)SC)nc(CNC(C2(C)CCCO2)=O)oc1C Cc1cnc(N)c(C(N2CC(C3(NC(=O)C=C4CCSCC4)CC3)C2)=O)c1 C1(NC(c2c(C)snn2)=O)CCCCC1NC(=O)CCOCc1ccccc1 C1(OCC(=O)NCC2CC2NC(c2n[nH]cc2C(F)(F)F)=O)CCCOC1 c1(C(N(CC(C)NC(=O)CCc2cn(C)nn2)C)=O)cc2cc(F)ccc2o1 c1(OCC)cccc(C(N2CCC(O)(C(C)C)C2)=O)c1N.C(=O)(CCCOC)N C(=O)(C(C(CC)CC)OC)N1CCC(NC(C(CCC)C)=O)C1(C)C c1(N(C2CCN(C(C3CCCC(=O)O3)=O)C2)CCO)ccc(Cl)cc1[N+](=O)[O-] c1(OC)cc(OC)c(S(=O)(=O)NC2COCCC2N(C)C)cc1OC c1(N(C)CCc2c(C)nccc2)cc(Br)ccc1S(=O)(=O)N1CCCCC1CF NC1CCc2ccc(NC(C3CC(O)C34CCC4)=O)cc21 c1(C(=O)NC2CC(OCC)C2SC)cccc(Cl)c1OC(C)C C(=O)(CCC(C)(C)C#N)N1CC2(C(NC(c3c(C)ncs3)=O)CC2)C1 c1(OC)ncccc1S(=O)(=O)N1CCCC(CCNC(c2cncnc2C)=O)C1 c1(OC)cncc(C(=O)NC(C)CC(C)NC(C2CN(C3CCCCC3)C2)=O)c1 C1(C(=O)NCCC(C)NC(C2(O)CCSC2)=O)CCN(c2ccc(Cl)nn2)CC1 N1(C(CCc2n(C)cnn2)=O)CCC(C(=O)NC2(C)CC3(CCC3)C2)=C(F)C1 c1(C(=O)NCC2C(NC(C3=CC(C)(C)C3)=O)COC2)ncnc2c1CCCC2 Cc1ccc(O)c(C(N2CCCC2CNC(C2CC3CCC2CC3)=O)=O)c1 C1(NC(c2cc(OC)ns2)=O)CCN(C(c2nnc(S)n2C)=O)CC1C C1(C(=O)NC2CC(N(C(=O)CCC3CCOC3)C)C2)CCC1(F)F C(=O)(C1=CC2CCC(C1)C2)N1CC2C(CC(=O)NCC3C(C)(C)CCO3)(CC2)C1 c1(C(=O)NC2(CNC(COCC)=O)CCOC2)cc2nccc(C(F)F)n2n1 C1(C(=O)Nc2cc(O)n[nH]2)(COC)CN(C(=O)CCc2nc(SC)no2)C1 C(C(C)CN(C)C(C1CCC1c1nc[nH]n1)=O)NC(COC(C)=O)=O C=CCC(C(=O)N(CCCN(C(=O)CC1CCOC1=O)C)C)NC(C)=O CCC(CCCC(=O)NC1C(C)C1C)NC(c1cc(C)cs1)=O C12(NC(CN3CC(=O)NC3=O)=O)CCN(C(c3cc(F)ccc3Cl)=O)CCC1C2 c1(OC(C(N2CCCCC(NC(CCCC=C)=O)C2)=O)C)ccc2c(c1)OCO2 c1(C(=O)NC2(COC)CN(C(C3(C(=O)OCC)CC3)=O)C2)ccc(=N)[nH]c1 C1(NC(CC2(C)CC2)=O)CC2CC(NC(=O)C=Cc3ccc(Cl)cc3)CC2C1 C(=O)(C(CC)C(=O)OCC)N(CC(CNC(C1CC(CCC)C1)=O)(C)C)C1CC1 C(C)(CCN=c1[nH]c(N(C)Cc2cc(Cl)ccc2Cl)nc2ccccc12)SC C(C(CC(C)C)C(=O)NCCCCN(C)C)NC(c1cc(CC)no1)=O C1(NC(c2ccc(Cl)cn2)=O)CC12CCN(C(C1CC3(C1)CC31CC1)=O)C2 c1(NC(N2CCC(O)(CCC(=O)N3CCCC3)CC2)=O)nc(Cl)c(Cl)c(Cl)c1Cl C1(NC(c2c(C)nco2)=O)CC2CCCC(C1)N2C(C1CN2CCC1(C)CC2)=O c1(C(=O)NC2CCN(C(=O)CN3CCCC3)CC2F)cc(F)c2ncccc2c1 N1(C(C(C2CC(C)(C)C2)OCC)=O)CC(NC(=O)CC2(CO)CCCC2)CC1C CC1CN(C(C2(n3cncn3)CC2)=O)CCN1C(c1coc(Br)c1)=O C1(C(N2CC(NC(c3cc(C)nn3C)=O)C(O)C2)=O)CCc2ncnn2C1 c1(OCC)nc(N2CC(CNC(c3cocc3C)=O)CC2C)ncn1 c1(C(=O)NC(CNC(C(CC)F)=O)CC)cnn(-c2ccc(O)nn2)c1CC N1(C(C(CSC)(C)NC(=O)Cc2sccc2C)=O)CCNC(=O)CC1 c1(NCc2scc(NC(C3N(C(C)=O)CC(O)C3)=O)c2)ccc2nnc(C)n2c1 C(C)(CCN(C)C(C1CC1(C)C)=O)NC(C1(COCC)CC1)=O Cc1ncc(NCc2ccc(C(F)(F)C(F)(F)F)s2)c(C)c1Br c1(C(C)(F)F)cccc(C(=O)NC2CCCC(NC(C3(CCF)CCC3)=O)C2)c1 c1(C(=O)NCC2C(C)(C)N(c3nc(C(F)(F)F)ns3)CC2)ccc([N+](=O)[O-])cn1 c1(NC(c2cccc(SCc3ccccc3)n2)=O)c(-n2cncn2)cccc1F C1(C(N(C2CCC(NC(=O)Cc3cnns3)CC2)C)=O)CCc2nccn2C1 c1(C(N(CCNC(C(CC)n2cncn2)=O)C(C)C)=O)ccc(C)nc1OC C1(CC(=O)NCC2CC2NC(=O)CC2CCOC2)CCC(CO)CC1 Cc1ccc(C(=O)N(CCCCC)C)n1C.C(=O)(C=CS(C)=O)N(CCCO)C Cc1ccn(CC(N2CC3CC3(NC(=O)C(C)(C)CC3CC3)C2)=O)c(=O)c1 C(=O)(CCCCCC#N)N1C(C=CC(=O)NC)CCC1 C1(F)(CNC(=O)CNC(C2CCCC2)=O)CCN(C(C2CC2C(N)=O)=O)C1 C=CCCC(C(=O)Nc1ccc(F)cc1CO)NC(=O)Cc1cc(C)nn1C C12(C(=O)NCc3c(C)nn[nH]3)CC(CCO1)N(C(=O)C(=O)C(C)C)C2 c1(SCC(=O)NC2C(NC(CCC3(C)CC3)=O)CCOC2)ccnc2c1CCO2 CN1CCC(C)(C(=O)NCCOCCCN(C)C(C2(F)CCCC2)=O)C1=O CC1CCc2[nH]nc(C(=O)NCC3CCCN3Cc3cc(F)ccc3F)c2C1 C1(CNC(c2cc(CCC)[nH]n2)=O)CC(C)N(C(=O)CCCCSC)C1 c1(C(=O)NCC(C)NC(C2OCCN(CC)C2)=O)cncn(C)c1=O c1(C(N(CCCOCCN(C(C(COC)(F)F)=O)C)C)=O)ccc(P(C)(C)=O)o1 C(N=c1[nH]c(=NCCCn2cnnc2CCO)c2sccc2[nH]1)C1C(C)C1 CC1Cc2ccc(C(=O)NC3CCCC(NC(c4nnn(C)n4)=O)C3)cc2O1 C1(C(N2CC(CNC(=O)CN3CCCS3(=O)=O)OCC2)=O)CCn2nnnc2C1 N1(C(CC2C(C)=NNC2=O)=O)CCN(C(C2CN(C3COC3)C2)=O)C(C)C1 c1(C(N(C2C(NC(C(C(CC)C)O)=O)CCCC2)C)=O)cnc2c(F)cccn12 N1(C(=O)CC2CCC3CC23)CCC2CN(C(C3CC4(CSC4)C3)=O)C2C1 C1(O)(C(=O)NC2C(NC(c3c(C)noc3)=O)CCCC2)CN2CCC1CC2 N1(C(CNC(C(CC)OC)=O)=O)CCCN(C(=O)C=Cc2ccncc2)CC1 c1(C(=O)O)ccc2c(c1)CCCN2C(=O)CC1(C(F)(F)F)CC1 N1(C(C2C(OC(C)=O)C2)=O)CC2(CC2)CC1CO.c12cc(c(C)o1)C(=O)NC2 C1(CNC(=O)CC2COCC2NC(c2ccc(C3CC3)o2)=O)CC2(C1)CC2(F)F C1(NC(C(c2c(F)cccc2F)(C)C)=O)C=CCC(C(=O)O)C1 C1(CNC(c2c(COC)ncs2)=O)CC(C)N(C(C2CCCOC2)=O)C1 c1(C(N(C(CNC(C=CCN(C)CC)=O)C)C)=O)cn(C2CCOC2)nc1C c1(C(N)=O)ccccc1C(=O)NC1CC(CCNC(C2CCC(F)(F)C2)=O)C1 c1(NC(C)=O)ccc(CC(=O)NC2CC2NC(=O)C(=C2CCCCC2)F)cn1 Cc1ccc(CC(=O)NCCCCCNC(=O)CCc2cncs2)c(Cl)c1 C1(C(=O)NCC2CN(C(CC(CC=C)(C)C)=O)CC(C)C2)CCc2nnc(C)n2C1 S(=O)(=O)(c1cccc(C)c1)N1C(C(=O)NC(C(=O)OC)Cc2csc(Cl)c2)CCC1 N1(C(CSC)=O)CCC2(CC1)CN(C(=O)CC1COCC1O)C2 C(=O)(C(C(C)C)C(C)C)NC1C(NC(CN(CC)CC)=O)COC1 C1(CSC)CCCN1C(=O)C(=O)NCC1(OC(F)F)CCCC1 C1(CCNC(C(c2cnn(C)c2)C)=O)COCCN1C(c1csc(Cl)c1Cl)=O N1(C(C=CCC(C)(C)NC(C(C)OCC#C)=O)=O)CC2CCCCC12C c1(C(N(CC(C)NC(c2c[nH]nc2F)=O)C)=O)cccc(NC(=O)N(C)C)c1 c1(NC(C(=O)OCC)=O)ncc(C(=O)NC(c2ccccc2)CN)cc1Cl C(=O)(N1CCN(C(=O)Nc2nc3c(s2)COCC3)CCO1)OC(C)(C)C NS(=O)(=O)C1(C(=O)NC2CCC(CNC(=O)CC3OCCO3)CC2)CC1 C1(NC(C(CC)SC)=O)CCN(C(=O)CCC(=O)c2ccc(OC)cc2)C1CC Cc1cc(C)c(S(=O)(=O)N2CCNC(=O)C2C(C)C)cc1-c1ccncc1 C12(NC(c3n(CCCC(=O)OCC)nnn3)c3ncco3)CC=CC(C1)OC2 C(=O)(CCCCCCn1cc(-c2nc(C)cs2)nn1)Nc1c(SC)cccc1 CCCC(C(=O)NC1CN(C(c2onc(C)c2C)=O)CC1CC1CC1)NC(C)=O c1(OC)nn(C)cc1C(C(=O)NC(C)C)N(C1CC(C2CC2)C1)C c1(OCC)ccc(F)c(C(=O)N(CCCNC(C2CC23CC3)=O)CCO)c1N C1(CC)OCCC1C(=O)NCCCCN(C)C(c1cncn1C1CC1)=O C(N=c1cc[nH]c(=NCCCc2ccccc2[N+](=O)[O-])[nH]1)c1nnc(CC)s1 C1(CNC(C(CCOCC)NC(C(C)OCC=C)=O)=O)CC2(CCC2)CO1 C(=O)(CCCCC(C)(C)OC)NC1CCCCN(C(CCCC#CC)=O)C1 CC1C(NC(=O)COC2CCCC2)CCN1C(=O)CCC1CCC1 c1(N2CCC(COCC)CC2)nc(N2CCC(CSC)C2)c2c(ncn2CC)n1 C1(C(=O)NC(CNC(C(CCC)CC)=O)(C)C2CC2)CCn2nccc2C1 C1(OC)COCCC1(c1nnnn1CC1CCOC1)Nc1cn(C)nc1OC C(=O)(C(O)C(F)(F)F)N1CC(C(N(CC(C)O)CC)=O)C(CC)C1 C1(CCN(C(C2N(C(C)=O)CCC2)=O)C)CCCCN1C(=O)C(C)=CC(C)(C)C CCCCC(C)CCC(=O)NC(C)(CC)CCNC(c1sccc1CO)=O CCCCCCC(CC)NC(C1COCC1NC(=O)C(C)NC(C)=O)=O N1(C(CSC(=N)N)=O)CCC(CNC(C2(C(O)C(F)(F)F)CCC2)=O)C(O)C1 C(=O)(C1=CCCCC1C)N1C(C(=O)NCc2ccc(C)cc2)CSC1 Cc1cn2c(CNC(=O)CC(C(C)(C)C)c3ccc(F)cc3)c(C)nc2s1 C(=O)(C1=NOC(C)C1C)NC1(C(C2CCCCC2)OC)CCN(C(CC)=O)C1 C(C(C)C(=O)NCC#CC(=O)NCC1C(C)C1C)OCC CC1(C)OCCC1C(=O)NC1(C(=O)NCC2(CC(N)=O)CC2)CCSC1 c1(CC(=O)NC2CCC(C)(NC(C3CNC(=O)N3)=O)CC2)noc2ccccc12 CN1CC(C(N2CCC(CCNC(c3cc(C(F)(F)F)c[nH]3)=O)C2)=O)NC1=O N1(Cc2c(C)nccc2)N(C)CCCC12CCCC2 c1(OCC(N2CC(NC(CCCOCC=C)=O)C2)=O)ccccc1C(F)F C1(N(CC(=O)NC2CCCCC2)C(C)=O)CCC(NC(C2CC2Cl)=O)CC1 C(=O)(C(C)(CC)CC)N1CC(CC)C(C(N2CCC(C)(C)C2C)=O)C1 C1(OCC(=O)N(CCCO)CCN(C)C)CCCOC1.C(=O)(CCOC)N(C(C)C)C C1(CNC(C2CCC(CC)C2)=O)CCCN(C(=O)CCc2ccc(Cl)nc2)C1 N1(C(=O)CCN2CCOCC2)CCCC(CCC(=O)Nc2cn3ccsc3c2)C1 c12ccc3cc(oc3c1)C(=O)N2.n1(C(C)C)nccc1CNC(=O)OC(C)(C)C Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)CCOc2ccc(F)cc2)C(C)C1)=O C(=O)(C(C)(C)C(C)(F)F)NCC1CCC(NC(Cc2cn(C)nn2)=O)CC1 N1(C(CN2CC(C)C2)=O)CCC(C)C(CNC(=O)Cc2nc([N+](=O)[O-])n[nH]2)C1 N1(C(CNC(Cc2cnc(C)s2)=O)=O)CCOc2ccccc2C1 c1(NC2CCCN(C(=O)CCN3C(=O)CCC3=O)C2)ncnc2cccc(F)c12 C(=O)(N(OC)C1CCC1)c1nc(CC(CCC=C(C)C)C)on1 CC1CC(C(=O)NCCc2ocnc2CNC(C2(F)CCCOC2)=O)=NO1 S(=O)(=O)(c1ccc(N)cc1F)NC(C)C(O)c1cccs1 C(=O)(C1CCc2nccn21)NC1CCN(C(c2c(N)cncc2)=O)C12CC2 C12(C(=O)NCC(C)O)CCCC(CCC1)C2O N1(C(CCC(CC)C)=O)CC(C)CN(C(=O)CCc2csnn2)C(C)C1 C1(C(N2CCOCC2CO)=O)CCCN(C(C2CCCC2CF)=O)C1 CC1(CCC(=O)NC2CC(CCNC(c3cncn3C3CC3)=O)C2)CC1(F)F C1(NC(=O)CC2CC(F)(F)C2)CN(C(C2CN3CCCC2C3)=O)CC2(CCC2)C1 C(CCC(C)CC(=O)NC1CN(C(c2nn(C)cc2C)=O)CC2(CC2)C1)=C(C)C c1(OC)ccc(CSCCC2(NC(c3cnn(C)c3C)=O)CC2)cc1.C1C(=O)N1 Cc1ccnnc1C(=O)NC(C)(CNC(=O)C(C)Cc1cccnc1)CO c1(OCC)cc(C(=O)NCc2ccn(C3CCCN(C)C3)n2)ccc1OC(F)F c1(NC2CN(C(C3CC(C(C)C)OCC3)=O)CC2(C)C)nc(Cl)nc2sccc12 c1(SCC(=O)NC(CNC(C(COCC)C)=O)CC)cc(=O)n2ccsc2n1 c1(C(N(CCNC(Cn2ncc(CC)c2)=O)C)=O)cc(C)c2[nH]nnc2c1 N1(C(CC2(C=C)CC2)=O)CCC(C2CCN(NS(N)(=O)=O)C2)CC1 C1(CNC(c2c(OC)ccs2)=O)C(C)CCN1C(c1[nH]cnc1C#N)=O C1(C2CCC2)(C(=O)NCC(c2cccc(Cl)c2)NC(C2(OC)CCC2)=O)CC1 C1(O)(CNC(CSCC=C)=O)CC2CCC(C1)N2C(=O)CC1CCN(C)CC1 N1(C(C(C=C)O)=O)CCC2(CC1)CN(C(=O)CN1CCNC(=O)C1)C2 C1(COC)(NC(c2n[nH]cc2Cl)=O)CCN(C(c2nc(C(C)C)oc2C)=O)C1 C12(C(N(CCOCCC(=O)NC(CC=C)CO)C)=O)CCC(C1)C2(C)C C1(Nc2cnn(C)c2-n2cnnc2)CC(P(C)(C)=O)CN(C(=O)OC(C)(C)C)C1 O=C(NN1CCCC1C(N1CCc2ccccc2C1)=O)C(F)(F)Br C1(C#N)(C(=O)NC(CC)CNC(=O)CC(C)COC)CCS(=O)(=O)CC1 c1(C(=O)NCCCN(C(CCC(C)C)=O)C)ccc(C(C)C)c(C#N)c1 N1(C(CCC=CC(C)C)=O)CC(CNC(=O)C(C)CN(C)C)OC2CCCC12 N1(C(c2ccc(OC)cn2)=O)CCCCC(CNC(=O)C(c2nc(C)cs2)C)C1 Cc1nc(-c2ccco2)cc(=NCCC(C)NC(c2ccc(CN(C)C)[nH]2)=O)[nH]1 c1(CN2CC3C(C(=O)NC4CCN(C)CC4)(C3)C2)cc(F)cc(Br)c1F c1(C(=O)Nc2cc(C)c(O)cn2)cc2ccc(-c3cnc4sccc4c3)cn2n1 c1(NC2(CNC(C3N(C(C)=O)CCC3)=O)CC2)cc(Br)c(F)cc1F C(=O)(C#CC1CCCC1)N1CCC(CC(=O)N(CC(CCC)C)C)C1 N1(C(c2cscn2)=O)CCCC(OCC(=O)C2CC2)C1 Cc1nc(C(=O)N(C(C)(C(=O)NC2CCC3(C(C)C)CC23)C2CC2)C)cc(O)n1 C1(CC(=O)NC2CC(C(F)F)(NC(C3CCCNC3=O)=O)C2)CCCC(F)(F)C1 c12ccc(cc1)[nH]c2=O.c1(CNC(C2(OCC)CCC2)=O)nc(NC(N)=O)co1 C#CCC(C)(CC)C(=O)NCC1CCCN1C(c1ccnc(OC(C)CC)c1)=O N(C(=NCCCC(F)F)N1CC2CCOC2C1)Cc1c(OC)c(Cl)ccc1 C12(COCC)CC(C(=O)Nc3ccc(N(C(=O)CSC(C)(C)C)C)cc3)(CO1)C2 N1(C(c2ccc(C(C)=O)[nH]2)=O)CCCC2(CNC(c3cncs3)=O)CC12 c1(OCC)ccc(N)c(C(=O)NCC2CN(C(c3nccn3C(C)C)=O)C2)c1 N1(C(c2ccn(COC)n2)=O)CCCC(C2CC2NC(=O)C2=C(Cl)CCOC2)C1 c1(C(N(CCN(C(C(C2CC2)OC)=O)C)C)=O)cnn(CCO)c1C(F)(F)F n1(CC)ncc(C(=O)N(C2CCCN(C(=O)Cc3c[nH]ccc3=O)C2)CC)c1C N1(C(COc2ccc(C)cc2)=O)C2CCCC1CC(NC(=O)C(C)(C)C(N)=O)C2 C(=O)(C1=CCCSC1)NCc1c(C(=O)NCc2cc(C)ncc2)occ1 C1(NC(c2cc(C)sc2C)=O)CCN(C(=O)C=CC(c2ccccc2)=O)C(C)C1 c1(OC)cnncc1C(=O)NC1C=CC(CC(=O)NCc2ncc[nH]c2=O)C1 c1(C(=O)NC2(C=C)CCCC2)cnn2cc(S(C)(=O)=O)cnc12 c1(C(=O)NC(C(=O)Nc2cn(C(C)(C)C)nc2)Cc2cn[nH]c2)c[nH]ccc1=O c1(CC(=O)NCC2C3CN(C(C=C(C#N)C#N)=O)C2C3)ccc(F)c(F)c1 CC(C)CCCCCC(=O)N1CC(NC(=O)OC(C)(C)C)C12CCC2 N1(C(CC(=O)NC2CC2)=O)CC2(CCN(C(=O)CC(c3cccc(F)c3)O)C2)C1 c1(OC)cc(Br)ccc1CN1CCC(CNC(c2ccc(F)nc2)=O)C1 CC(CCCCNC(c1ccc(N(C)C)[nH]1)=O)NC(=O)CCN(S(C)(=O)=O)C c1(CN2C(=O)CC3C(C3)C2)cnn(C(=O)NCC)c1.C1(CC)CC1(C)C C1(CNC(c2csc(N3CCCCC3)n2)=O)C2CC2CN1C(=O)C1=CCSC1 Cn1cnc2cccc(C(=O)NC3CCC4(CC3)CN(C(C35CC(C3)C5)=O)C4)c12 C(=O)(CC1=CCOCC1)NC1CC(OC)CN(C(C(CCCC)O)=O)C1 c1(CCC)nc(C(=O)NCC(C(C)C)NC(=O)C(O)C2CCC2)co1 Cn1c(C(=O)NCC(C)(C)NC(=O)COCC2(F)CC2)cnc1Br c1(NC(CC(C)NC(c2ccn(O)c(=O)c2)=O)C)ccnc2ncnn12 CC1CCC(=CC(=O)N(C(CNC(=O)C(C2CC2)N(C)C)C2CC2)C)CC1 C(CCN=c1ccc(S(=O)(=O)NC2(CO)CCSC2)c[nH]1)(C(C)C)OC C1(NC(CC2(COC)CC2)=O)CC(O)CN(C(=O)Cc2ccnc(C)c2)C1 C(C(CCOC)NC(C1CC2CC2C1)=O)NC(CCC)=O c1(C(N(CCn2cc(-c3n(CC(=O)OC)ccn3)nn2)C)=O)nnc(O)cc1C C1(CN(C(COCc2cc(C)no2)=O)C)CCCN(C(=O)C(C)(C)O)C1 N1(C(C)=O)CCCCC(NC(C(CC)CC)=O)C1.C1(=O)C(C)(c2ccccc2)N1 CCCC(O)CC(=O)N(C)CC1(CNC(c2cnc(Br)c(N)n2)=O)CC1 c1(C(=O)OC)cc(CO)cc(NC(N2CCN(C(=O)Cc3cccs3)CC2)=O)c1C N1(C(CCC#C)=O)CC2C(CNC(=O)C(c3ccc(OCC)cc3)C)C2C1 c1(C(=O)NC2CCCC(NC(c3ccc(CO)o3)=O)CC2)ccn2nccc2c1 c1(OC)c(C)nc(C2CC2)[nH]c1=NCCCC(C)NC(c1nnc(C)s1)=O N1(C(C2(C#N)CC=CC2)=O)CCC2CC2(NC(=O)C=Cc2cccs2)CC1 C1(C(=O)NCC2(COC)CCCO2)(C(C)C)CCN(C(=O)C(C)NC=O)C1 C1(NC(C(OC)OC)=O)CC2CN(C(C3(C)CCN(C)C3=O)=O)CC2C1 N1(C(c2cccc(OC)c2F)=O)CCC2(C1)CN(C(=O)C(C)(O)C(C)C)CCO2 C1(CCC(N2C(CNC(C3(CC)CC3)=O)CC2)=O)CCCOC1 CCC(C)C(=O)NCC(=O)NCC1(C)CC(NC(c2cc(C)c[nH]2)=O)C1 C1(NC(C(F)=CCC)=O)CCCC12CCN(C(=O)C=CCCC)CC2 CC1CN(C(C2CNC(=O)CC2(C)C)=O)CCCN1C(c1csc(CO)n1)=O c1(C(=O)NC2CC23CC(NC(=O)CCCN2CCCC2)C3)c[nH]c2ncccc12 c1(C(=O)NC(CNC(C(C)OCCN(C)C)=O)CO)cc(Cl)c(F)cc1F N1(C(C(C)O)=O)CC(CO)C2(C1)CN(C(c1cc(P(C)(C)=O)ccn1)=O)C2 N1(C(C)=O)CC(NC(c2ccc(NC(c3cc(CO)no3)=O)nc2)=O)C(C)C1 CC(C)CC(C)(O)C(=O)N1CC2CCC1CN2C(C1CCCC1C1CC1)=O C1(C(=O)NCC2CC(CNC(C(C)c3cccs3)=O)C2)CCCN1S(=N)(=O)N(C)C N=c1[nH]nc(C(N2CC(O)(CCNC(=O)Cc3cncnc3)C2)=O)[nH]1 C=CC(C)(C)CC(=O)NCC1CCN(C(=O)Cc2ccc(C(F)F)cc2)C1 C1(CCC)CN(C(=O)C=C(Cl)Cl)CCN1C(C1CC1(C)C(F)(F)F)=O c1(C(N2CC(CNC(C3CCO3)=O)OCC2)=O)cccc(O)c1Br C1(C(=O)NCCn2ccc(C)n2)CCCCC1NC(=O)CCOC(C)C N1(C(C=CCC)=O)CCC(N(C(=O)C2=CCCC2)CCO)CC1 N1(C(C(C2CCOCC2)OCC)=O)CCN(C(c2ocnc2C)=O)C(C)C1C c1(C(N(CCNC(c2nc(SC)oc2)=O)C)=O)cnc(C(N)=O)c(Cl)c1 C(=O)(C1=C(Cl)CCC1)NC(C(=O)NCC(N1CCCC1)C)C1CCCC1 C1(O)(CNC(C(C)SCc2ccccc2)=O)CN(C(=O)C(C)(C)O)C1.C1(=O)CN1 C(C1c2ccccc2CCN1CC(=O)NC(N)=O)NC(=O)CCCC1CCCC1 c1(C(=O)NCCC2CCN(C(C3CC4CCC(C3)O4)=O)C2)c(F)ccc(Cl)c1F c1(SC)cc(C(=O)NCC2CCN(C(C3CCCCO3)=O)C2(C)C)ccc1N C1(CC(=O)N(C2(C(N3CCC(Oc4cn(C)nc4)C3)=O)CC2)C)CC2COCC12 C(=O)(C(C)(C)CCCNC(c1ccccc1C#N)=O)NC(C(C)C)CN(C)C c1(C(=O)NC2CC(CCNC(C(CNC(C)=O)(C)C)=O)C2)cc2cscc2s1 C#Cc1cncc(C(N2CCC(c3ccc(NC(=O)CNC(N)=O)cc3)C2)=O)c1 C1(NC(=O)C=CC2CC2)CC(C2CCN(C(=O)Cc3ccc4nn[nH]c4c3)C2)C1 c1(C(N2CCC(N(C(=O)CCCCCN(C)C)CC)C2)=O)ccc2sncc2c1 c1(C(=O)NCC2N(C(CSCCOC)=O)CCCC2C)ccc2c(n1)CCCC2 CCCCC(=O)C(=O)NC1CCC1CNC(=O)CCn1nc(C)nc1C c1(-c2nnc(N3CCC(OCC)C3)n2CC(C)OC)cccc(Cl)c1Cl C#CC1(c2ccccc2)CN(C(=O)C(c2cc(Br)no2)=O)C1 C#CCC(C)(CC)C(=O)NCc1cncc(C(=O)NC(C)CC(=O)OC)c1 C1(C)(CNC(CCOCC#C)=O)CCCN1C(C1COCCOC1)=O Cc1cc(C(N2CCOC3(C2)CN(C(=O)CC2(O)CCC2)C3)=O)cc2c[nH]nc12 N1(C(CC2(C)N(C(C(C)c3ccsc3)=O)CC2)=O)CCOC2COCC12 c1(C(=O)OC)cnc(CNc2ncc(Br)c(Br)n2)c(F)c1 C(CN=C(NCCF)N1CCC2=NC(O)=C2C1)C1C(C)(C)C1(Cl)Cl c1(C2C(C)(C)C2C(=O)NCc2ccn(-c3ccncc3)n2)cc(Cl)c(Cl)cc1N CC1CN(C(c2cnnc(-c3ccccc3)c2)=O)CCN1C(C1(F)CCOC1)=O C#Cc1ccccc1NCc1cccnc1OCC1CC1 CCC(C)C(C(=O)NC1CCCN(C(C)C)C1)N(C(=O)CC1CCCCO1)C C1(NC(COC(C)(C)C)=O)CCN(C(=O)C(c2ccc(F)cc2)(C)F)CC1CO c1(-c2ccn3ncc(OC)c3c2)nc2c(s1)CN(S(CC=C)(=O)=O)CC2 N1(C(CN(C2CCS(=O)(=O)C2)C)=O)CCOC(CNC(=O)CSCC2CCCO2)C1 O=C1CCCCC(C(=O)NC2(C(=O)NCC3CC(C4CC4)=NO3)CSC2)N1 N(C1c2ccccc2CC1NC(C1C(C)C1(F)F)=O)C(C(CC)n1cncn1)=O c1(NC(CC(C2CC2)NC(CC(CC)(F)F)=O)=O)ccc2occc2c1 N1(C(CNC(=O)OCC)=O)CCC2(CC1)CC(NC(=O)C(F)CC1CCOC1)C2 CC1CCN(C(C2CCCN2N=O)=O)CC1N(C(=O)CCc1ccc(Cl)cc1)C N1(C(CNC(=O)OCC)=O)CCCCC(NC(=O)CCc2cncs2)C1 Cc1cn2c(n1)CC(C(=O)NC(C)CNC(C1(CN(C)C)CC1)=O)CC2 N1(C(c2ccn(C)c2)=O)CCN(C(=O)CCc2cccn2C)C2CC12 c12ccc(c(OC)c1C)C(=O)C2N(C(CC)CO)C.C1(N)CCC2(CC1)CC2.OC c1(CC(N2CC(O)(CNC(C(C)C3CCCO3)=O)C2)=O)ccc2n[nH]cc2c1 C(C)(C1OCCc2sccc21)NC(=NCCCOC)NCC(C)(C)C(C)(C)O C1(C(=O)NCCC2(O)CN(C(C(C)c3cc[nH]n3)=O)C2)CCc2ccccc2C1 O=C1CCC(CN(N2CCOC(C(F)F)CC2)C(c2ccc(F)cc2)=O)C(=O)N1 C1(NC(c2cccc3ccnn23)=O)CC2CCC1C1CN(C(=O)CSC(F)F)CC21 N1(C(C(F)=CCC)=O)CCC(C(F)(F)F)C(NC(=O)CCCCOCC)C1 C(=O)(CCCCC#N)N(C)CC(=CC(=O)NOCCCF)C1CCCC1 c1(C(N2CC(C)N(C(=O)C=CBr)CC2)=O)ccc2c(c1)[nH]c(=O)[nH]c2=O C(=O)(C1CSc2ccccc21)N1CC(C)C(CNC(=O)CCC2CC2(F)F)C1 C(C)(C)(CCC(=O)NC1CCC(NC(=O)CCc2ncc(C)[nH]2)CC1)OC C1(NC(c2cccc(C(C)C)c2)=O)CCC(C)N(C(=O)CCN2CCOCC2)C1 C1(CNC(C(C(C(C)C)OC)O)=O)CCC12CCN(C(C1CCC(=O)N1)=O)CC2 C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1C(NC(Cn2ccc(C)n2)=O)CCC1 C1(c2nnnn2C)(CC)CN(CC2(N)COCCN2C)CCS1(=O)=O CCC(CC1CCCC1)C(=O)NC1CCCC1CNC(=O)CC(F)(F)F Cc1nc2cccc(C(=O)NCC3CC4COCC4N3C(=O)C=C(Cl)Cl)c2[nH]1 Cc1cccc(C(=O)NC2CCN(C(=O)CN3CCCC3CO)CC2CO)c1F c1(OC)ccc(CC(=O)NC2CCC(NC(c3cnoc3C)=O)C2)cc1 c1(C(N(CC(C)C)C(c2c(CC)scc2)=O)=O)cc([N+](=O)[O-])cc(C)n1 C1(Nc2cccc(I)c2O)COCCN(C(c2cnc(N(C)C)nc2)=O)C1 C1(C(=O)NCC(C2CC2)NC(C2CC3(CCC3)C2)=O)CC2(CCCCC2)C1 S(=O)(=O)(c1cccc(F)c1)N1C(C(=O)Nc2cnn(C(F)(F)F)c2)CC1 C#Cc1ccnc(C(=O)NC2CCCC2NC(c2nc(Br)c[nH]2)=O)c1 c1(CC(C)C)cn(CC(=O)N(C)CC2CCOC2C(=O)O)nn1 CCCCC(O)C(=O)NC(CO)C(C)NC(c1cc(-n2cnnc2)ccn1)=O N1(C(C2CCC(CCC=C)C2)=O)CCC(c2ccc(CO)cc2)CC1 N1(C(c2c(C)nn(C3CC3)c2)=O)CC2(CC2)CC1CNC(=O)CC1COC(=O)C1 c1(C(=O)NC(C(=O)N(C)CC2CC(O)C2)Cn2ccnn2)c[nH]c2nccc-2c1 C(=O)(C1CSc2ccccc21)NCC12OC(C)C(NC(=O)CC3CCC3)(C1)C2 Cc1cc(N)c(C(N2CCC2CNC(c2c([N+](=O)[O-])cnn2C)=O)=O)nc1C c1(C(N2CC(OCC(N3CCC(OCC(N)=O)C3)=O)C2)=O)ccc(O)cn1 N1(C(C2(CC#C)CCN(C(C3CC34CC4)=O)C2)=O)CC(CC)CC(C)C1 C(=O)(C1=NOC2(CCC2)C1)NCC(CCC)C(=O)NC(c1ccccc1)CO S(=O)(=O)(c1cccc(-c2cccc(CC(=O)NC(CC3CC3)CO)n2)c1)NC C1(NC(c2occ(C)c2)=O)CN(C(=O)CC(c2c(C)noc2C)C)CCC1(C)C C12(CNC(c3cc(C)sc3C)=O)CCC1CCN2C(=O)C(c1cccn1C)=O n1(CCC)c(CCCCNCc2sc(Cl)cc2Cl)noc1=O c1(C(N2C(C(C)NC(=O)OC(C)(C)C)C(C)C2)=O)ccc(SCCCF)cc1 C(CCCCC(=O)N(CCCC(O)CO)C)NC(c1cnc(CC)nc1)=O C1(C(=O)NC2(CC(=O)NCCC3(O)CCCC3)CC2)CCC(C2CC2)C1 c1(C(=O)NC2CCN(C(c3c(C)con3)=O)C(C)C2)cc(F)c(Br)cc1F CC1CC(NC(=O)COCC(F)(F)F)CCN1C(c1nnn(C)n1)=O c1(C(=O)NCCN(C)C(c2cnc(C(F)(F)F)nc2)=O)cc(Cl)c(F)cc1O C#CC1COCCN1C(c1ccc(-c2cccc(Br)c2C)s1)Cc1occc1Br c1(CN(CC(c2cn(CCOC(C)=O)nc2)=O)C)cc(Cl)c(Cl)s1 c1(C(=O)NC2C(NC(C3(C#C)CCCC3)=O)CCOC2)cccc(S(C)(=O)=O)c1 c1(OC)cccc(CN2CCC(c3nc(C(F)(F)F)cs3)C2)c1OC(F)F C1(NC(C(F)=CCC)=O)CCCN(C(c2ccn(-c3cccc(N)c3)n2)=O)C1 C1(C(NNC(=O)NC2C(C)OCC2)=O)CCC(C#N)C1.C(=O)O C12(NC(CCC=CC(C)C)=O)CCC(CC1NC(=O)CC(=O)N(C)C)C2 Cn1cc(OCc2csc(-c3ccncn3)n2)cn1 c1(OCCNC(c2ccc(OC)cc2)=O)cc(C)ccc1C C(=O)(C1COc2c(F)cccc21)N(CC(C)(C)O)Cc1c(OC)cccc1 C(=O)(CCC(C)C#N)N(CCCCCNC(C=CC(C)C)=O)C c1(CCOC)ccc(S(=O)(=O)Nc2ncncc2C(N2CCC(C)(O)C2)=O)cc1 N1(C(c2c(C)cc(SC)s2)=O)CCC2CCN(C(=O)CC(C)(C)N(C)C)CC12 c1(C(=O)NCC(CO)NC(C2CC(F)(F)C2)=O)ccc(=NCC2CC2)[nH]c1 c1(C(N2CCCC(CNC(C=COCC)=O)CC2)=O)ccnc2[nH]c(C)nc12 c1(C(N2CC(C(N3CCC(O)C(O)C3)=O)C2)=O)c(OCC)nn2ccccc12 C1(C2CC2)(NC(C2N(C(c3cc(C)c(N)cn3)=O)CCOCC2)=O)CCCCC1 N(C1COc2cc(Br)ccc21)CC1(OC)CC2CCC1CC2 N1(C(C=C(C)C)=O)CCC2(CC1)C(NC(=O)C=Cc1cc(Cl)ccc1Cl)CS2(=O)=O CC(C)(CCCNC(c1ccc(C#N)cc1)=O)C(=O)NCCc1cscn1 N1(C(c2ccc(OCCC)cc2)=O)CCN(C(=O)CC=C(Cl)Cl)CC1C(C)C C(=O)(C(C(C)CC)NC(c1cccc(Cl)c1C(F)F)=O)NC(CC)CNC(C)=O c1(NCC(=O)N(C(c2ccccc2)C)C)cc(F)ccc1-n1nccn1 CC1CN(C(=O)CN2CCCC2=O)CC2(CCN(C(C3CCCSC3)=O)C2)O1 CCC(CC)C(F)C(=O)NCC1(C)CCCN1C(C1CCS(=O)CC1)=O C1(CNC(c2cc(CC)no2)=O)CN(C(c2cccc(C)c2N)=O)C2CCN1C2 c1(N2CC(CN3C(c4n(C(C)C)ccn4)CCC3)C2)cc(F)c(N)c(F)c1F c1ccccc1C=CC.n1(C2(OCCC)CC2)cc(C2(O)CCOC2)nn1 C1(N(C2CCC2)CC2CN(C(N(C)C)=O)C2)=CN=COC2=CC=NC2=N1 c1(C(=O)Nc2nc(OCC)c(Br)cc2)cn2c(C)ccc(-c3cnn(C)c3)c2n1 N1(N2C(C(C3CCCCC3)C)CC2)CC2CCC(C2)C1=O Cc1cc(NC(c2ccc(C3CC3)o2)c2nnnn2C(C)(C)C)ccc1[N+](=O)[O-] c1(N2CCN(CCNC(c3c(SCC=C)cccc3)=O)CC2)ncnc(Cl)c1F N1(C(C(COC)OC)=O)CCOCC(NC(C2(C)CCCC2C)=O)C1 CCCCC(C(=O)NC1CCC1NC(c1c(C)oc(C)c1C)=O)C(C)C C1(CC(=O)NCC2(F)CCN(C(=O)C(F)C3CCC3)CC2)CC2(CCCC2)CO1 CCCC(C(=O)N1CCC(C2CC2)C1C(=O)NOCC1(C)CC1)C(C)C c1(CC(C(=O)OC)NC(=O)C(CO)N(C)C)ccc(F)cc1 C1(C(N2CC(N(C)C)(C(N)=O)C2)=O)CC(C)(C)CN1C(=O)CC1CSCCO1 C1(C(=O)NCCC2N(C(CC3CC(=C)C3)=O)CCCC2)CN2CCCCC2CO1 N1(C(C(C)NC(c2ccccc2)=O)=O)CCOCC1CNC(=O)CCS(C)=O c1(OC)nc(C)ncc1C(=O)NC(CNC(=O)Cc1n[nH]c(C)n1)C1CCC1 N1(C(C2(CNC(C3C(C#N)C3)=O)CCCC2)=O)CCC(O)C(F)C1 c1(OCC)ccc(CCC(=O)N(CC(O)CN(C)C(c2cnsc2)=O)C)cc1 C(=O)(CCC(F)(F)C(F)F)NC1CN(C(COC(CC)C)=O)CC(O)C1 C1(NC(CCOC2CN(C(C(C)SCCCC)=O)C2)=O)CCCC(N(C)C)C1 C1(CC=C)(NC(C2CC(O)(C#C)C2)=O)CCCN(C(C2CN(C)CCO2)=O)C1 c1(SC)ccc(N)cc1C(=O)NC1COCCC1NC(C1CCC(C)O1)=O N1(C(COCCC)=O)CCCC(N(C(=O)C(C)SC)CC)C1 C1(C2N(C(COC(C)(C)CNC(C3CCN3C)=O)=O)CC2)CCCCC1 N1(C(c2ccc(C(=O)OC)nc2)C(=O)NCCC2CC2)CC2COCC2(C)C1 C(=O)(C(CC(F)F)NC(c1ccoc1)=O)NC1C=CC(C(=O)OC)C1 C1(CC(=O)NC2(C3N(C(CCC4N(C)CCC4)=O)CCC3)CC2)CCC2CC2C1 C#Cc1ccc(F)c(C(N2CCN(C(=O)C(C3(O)CCCC3)F)CC2C)=O)c1 C1(C)(NC(c2n(CCC)ncc2)=O)CCN(C(=O)CNC(c2cccs2)=O)C1 N1(C(N2CC3CCCCC3(CC(=O)OC)C2)=O)CCC2(CC1)COCCO2 C(=O)(C(C(C)N(C)C)C(C)C)NCC(CNC(CCn1c(=O)sc(C)c1C)=O)C C(=O)(CCC(C)CN(C)C)NCc1nc(CNC(c2nncc(OC)c2)=O)sc1 N1(C(CCN(CC)CC)=O)CC(NC(C2CC2[N+](=O)[O-])=O)C(C)C1 c1(C(=O)NCCC(C)NC(c2nc(CCC)oc2)=O)cc(F)cc(S(N)(=O)=O)c1 c1(NC(CC#C)=O)cc(C(N2CCC(c3ccc(F)cc3)CC2)=O)n(C)c1 CCC(CC(F)F)C(=O)N(CCCOCCN(C(=O)Cc1ncoc1C)C)C c1(C(=O)NCc2ccc(CNC(=O)C=Cc3ccco3)cc2)cn2c(n1)CCC2 CCC(CC(=O)N1CCCC1CN(C(=O)CCc1ccc[nH]1)C)C(C)(C)C c1(C(=O)NC(C)C(=O)NCC(F)F)cc(O)cc(F)c1.C1(c2cccs2)C(=O)N1 c1(C(N2CCC(N(C)C(C3CC(C4CC4)=NO3)=O)C2)=O)ccc(N=[N+]=[N-])cn1 C1(C2CCN(C(c3cc4c(F)cccc4[nH]3)=O)CC2)(NC(=O)C2=C(Cl)CC2)CC1 Cn1ccc(CNC(C2(NC(c3cnc(N)cn3)=O)CC(O)C2)=O)cc1=O c1(C(=O)NC(CC(C)NC(c2c(C)nc(C)[nH]2)=O)C)cc(Cl)c(Cl)n1C c1(NCC2CCCCN(C(C(C)=C(C)C)=O)C2)cc(=O)n(C)c(O)n1 C1(C(N2CCC(N(CC)CC)CC2)=O)CN2CCN1C1CN(C3CC3)CC2C1 Cc1[nH]nc2ccc(C(=O)NC3(C(N4CC(CNC(N)=O)C4)=O)CCCC3)cc12 c1(C(N2C(CC(=O)Nc3c(C)nccc3)CCC2)=O)cc(-n2cccc2)cc(Br)c1 N1(C(=O)OC(C)(C)C)CCCC2C(CC(=O)NC3(CCCF)CC3)C(C)(C)C12 c1(C(=O)NCC2N(C(CC(=O)NCC#C)=O)CCC2)c(OC)ncc(Cl)c1C c1(Cc2c(C3CN(C(=O)OC(C)(C)C)C3)nsc2N)cc2cccnc2[nH]1 C1(C(N2CC(C)(OCC(=O)NCC(C)(C)C#N)C2)=O)CC1C1CCCC1 c1(C(=O)NC(C2CN(C(=O)CCNS(C)(=O)=O)CCO2)C)cnn2ncccc12 C12(C(=O)NCC3CCN(C(COCCCC)=O)C3)CCC(O)C1CC2 N1(C(C2(NC(C(=O)N(C)C)=O)CSC2)=O)CCc2nnn(C)c2C1 C(=O)(N1CC(C)(O)CO1)C1CCN(C(c2cc(C)c(O)nn2)=O)C1C C1(OCC=CC(N2CC(N(CC)CC)C2)=O)CCOC(=O)CC1 C1(CC(=O)OC)CN(C(=O)Nc2cnc(O)c(F)c2)C2COCC2O1 Cc1c(C(=O)NC(C)(C)C(C)NC(c2cc(F)c(F)c(F)c2)=O)cc(O)cc1N C1(C#N)(C(=O)NC(C2(CNC(=O)CCc3c(F)cccc3F)CC2)C)CC2CC2C1 C1(C(=O)NC(CC)C(=O)NC2CCCN(C(C)C)C2)Cc2nccn2C1 C(=O)(C1=NOC(NCCCOCCCNC(c2ccc(=O)n(C)c2)=O)C1)OC C1(NC(=O)C(F)CC2CCCC2)CC(N=c2nc(CC3CCCCC3)[nH]s2)C1 N1(C(C(C)(C)OC)=O)CC=C(CC(=O)NC(C)C(=O)NO)CC1 N1(CC)CCC(F)C(C2OCCC2Sc2cccc(CNCc3nn[nH]n3)c2)C1 c1(C(=O)OC)cccc(NC2CN(C(=O)CC(C)SC)CC2(C)C)c1[N+](=O)[O-] C1(C(N(CC(CC)NC(=O)Cc2cccs2)CC)=O)CC2(CO1)CC(F)(F)C2 Cc1[nH]nc2ncc(C(=O)NCCNC(=O)CC3CCOC3)cc12 CC(C)(C)CCCCC(=O)N1C2CCC1CC(F)(CNC(c1nccs1)=O)C2 c1(OC)cnc(F)cc1C(=O)NC(C)CC(C)NC(C1(CO)CCC1)=O CS(=O)(=O)c1cscc1C(N1CC(CNC(c2cc3n(c2)CCOC3)=O)C1)=O c1(CC(C)C)nnc(NCC2CCC(NC(=O)C(C)(O)C3CC3)C2)s1 N1(C(c2n(CC)ncc2)=O)CC2CCCC2(NC(c2ncccc2Br)=O)C1 C1(NC(C(CC)F)=O)CN(C(=O)COCc2nc(C(C)C)no2)CCC12CCC2 C(=O)(C(CSC)N(C)C)NCCOCCNC(C=C(CC)C)=O Cc1cnncc1C(=O)NCCC1CCC(NC(=O)C=Cc2ccncn2)C1 N1(C(c2c(OC)nccc2)=O)CCCC(NC(=O)Cc2cc(C)ns2)C1C C1(CNC(Cn2nnc(C)n2)=O)CCCN(C(C2CCCN(C(=O)CO)C2)=O)C1 C#Cc1cnc(C(N2CCCC2c2cccc(C)n2)=O)c(C)c1 c1(OCC=C)ccc(-c2nc(CC)nn2CC2CCCCC2)cc1OCC c1(CCCC)cc(C(=O)NC2CC(CCNC(C3(C)CS(=O)(=O)C3)=O)C2)c(C)o1 Cn1cccc1C(=O)NCCC1CC(NC(C2CC(C)(C(C)(C)C)C2)=O)C1 C1(CC)CN(C(c2ccc(Cl)s2)=O)CCN1C(C1CCN1C)=O c1(N(CCOC)CC2CC(F)(F)C2)cc(Cl)nc2c(C)cnn12 CCCCC(F)C(=O)N1CC2C(CC(=O)NCC3CC(SC)C3)C2C1 C1(NC(c2ccc(OC)nc2)=O)CCC(C)N(C(c2c(C)cccc2C)=O)C1 CC1(C)CC=C(C(=O)NCC2(NC(=O)Cc3cc(Cl)sc3Cl)CC2)CC1 C1(C(N(CC(C)NC(C(CC(=C)C)OC)=O)CC)=O)CCCCC(F)(F)C1 C1(C(=O)Nc2c(C)ccc(CO)c2)CN(C(=O)C2=COCC2)CC12CCC2 C1(C(=O)NCC2(O)CC(NC(C(C)(C)OC(C)C)=O)C2)CCC([N+](=O)[O-])CC1 C(=O)(C1=CCOC1)N(C(C)CCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O)C c1(C(=O)NCC(CC)NC(=O)Cc2cscn2)ccc(CSC(F)F)o1 N1(CCC(=O)NCC(CNC(C2(C(=O)NC)CCC2)=O)F)CCOCC1 c1(C(N2CCC3(NC(c4csc(CO)n4)=O)C(C2)C3)=O)nccc2occc12 c1(COCC(=O)NCC2CN(C(=O)COC3CC3(F)F)C2)ccccc1Cl C(N=c1nc(-c2ccsc2)c(F)c[nH]1)C1CCN(C(C(C(CC)C)C)=O)CC1C c1(OCC)cccc(NC(=O)NC(CC(=O)OC(C)(C)C)CC)c1 Cc1nn(C(C)C)c(C)c1C(=O)NCCCC1CCCN1C(C1CCOCC1)=O C1(CCNC(c2cc(F)c[nH]2)=O)CN(C(=O)CC2CCCS(=O)(=O)C2)CCCO1 C#Cc1cccc(C(N2CCC(F)(CNC(C3CN(C(=O)N(C)C)C3)=O)C2)=O)c1 CC1CCC(=O)N2CCN(CC2)C2CCCN(C2)C(=O)CO1.c1(C)nc[nH]n1 c1(CC)nccn1CC(N1CCC(C(C)(C)NC(=O)CN2CC(C)(OC)C2)C1)=O C(=O)(C1=CCCOCC1)N(CCCCCNC(c1cccnn1)=O)C Cc1ncc(C(=O)NCCCC2(NC(C3CC(C)CCO3)=O)CC2)c(C)n1 C1(NC(C2C(OC)CCC2)=O)CCN(C(C2CN3CCN2CC3)=O)CC1F c1(SC(C)C)ncccc1NC(=O)COC1CC(NC(C2CC2(F)F)=O)C1 CC(C)C(CCNC(=O)C(C)CSC(F)(F)F)NC(=O)CC1CCCO1 c1(C(N2CCN(C(C(CC)C)=O)CC2C2CC2)=O)ccc2nnnn2c1 S(=O)(=O)(c1cccnc1NCc1cncnc1)NCC1(P(C)(C)=O)CC1 c1(C(=O)NC(C2CN(C(C(CC)(C)CC)=O)C2)C)c(F)ccc(OC(F)F)c1F N12CCCCC1CC(C)C(OC)=CC=NC=CC2=O C1(NC(=O)NC(C(=O)OC)C)CN(C(C2CCN(C(C)C)CC2)=O)CCC1F N#CC1(C(=O)NCC2CC(NC(c3ccc(CO)c(F)c3)=O)C2)CCCOC1 C1(N(C(=O)CC2CCOC2)C)CCC(NC(c2cnc(C(F)(F)F)cn2)=O)CC1 C1(NC(c2c(C)ocn2)=O)CCCCC12CCN(C(C1CCC(C)C1)=O)CC2 N1C(=NCC2CC(F)(F)C2)N2CCCC(C2)C1.CC1CCN(C(N)=O)C1 C(CCC1CC1)(C(=O)NOC(C1CCCO1)C)NC(=O)CC(=O)NCC#C CC1CCC(NC(=O)C(F)(F)c2nccn2C)CN1C(C1CCOCC1)=O N1(C(C2CC23CCN(Cc2cccnc2)C3)=O)CCC2(CC1)OCCO2 C1(C(N(C2(CNC(CC(=O)NCC)=O)CC2)C)=O)CCC(C)(C)CC1 C1(NC(C(C(C)(C)C)CO)=O)CCC12CCN(C(c1ccoc1)=O)CC2 C(=O)(C(C1CCCO1)C1CN(C(c2nccs2)=O)C1)OC.C1(=O)C(C)N1 c1(OCC)ccc(C(=O)NC2CNCCC2(F)F)cc1[N+](=O)[O-] C1(CN(C(C(C2CCC2)OCC)=O)CC)CCCCN1C(c1ocnc1C)=O C1(C(=O)NCCCC2CC(C)C2)CCCC(NC(C2(C(C)(F)F)CC2)=O)CC1 CC1COCC(C(N2CCOCC2CC(N2CC(S(C)=O)C2)=O)=O)O1 C1(CNC(CCCC#C)=O)CN(C(c2cnc3[nH]cncc2-3)=O)CCC12CCC2 CC(Cn1ccnc1)CN=C(NCc1ccccc1)N(C)CC(C)(O)C1CC1 Cc1ncc(C(N2CC(O)CC2C(N2CCCC2(C)C(N)=O)=O)=O)cn1 C1(c2nc3cccc(C)n3c2)CCN(N2CCCC(CO)(CO)C2)CC1 C(=O)(CCCC(=O)NC1(C)CC(CNC(=O)CC(C)F)C1)N(CC)CC C(CCCCCCCC(=O)NC(C)CCNC(C1CSCCS1)=O)(OC)OC c1(C(N2C(C)CC(CNC(=O)COC3CCC3)C2)=O)cc2nc[nH]c2cc1F C1(C(=O)NCC2N(C(CN(C(=O)OC)C)=O)CCC2)CC2CCC1C2 C#Cc1cc(F)c(C(N2CC3CC3(NC(=O)C(C)(C)c3ccno3)C2)=O)c(F)c1 CCCCC(O)CCC(=O)N1CCC(C(C)NC(C2NC(=O)CC2C)=O)C1 CCCC(C)CC(=O)N1CCCCC1c1n[nH]cc1C(N1CC(C#N)C1)=O CCC(O)(CC)CCNC(C1(C)CC1C(F)(F)F)=O C1(CC)(OC(=O)CC2CN(C(c3ccccc3)=O)C2(C)C)CCCCC1 Nc1cc2c(cc1C(=O)NC1CC1NC(c1ccc(Br)cn1)=O)OCCO2 C(=O)(C1CCCc2cncn21)N1CC(C(C)NC(=O)COc2ccccc2Cl)C1 CCC(CNC(=O)C(CC)CCOC)(CC)C(=O)NC1CCC1(C)C c1(C(=O)NC2CC(CNC(c3cc(C#N)ncc3)=O)C2)oc2ccccc2c1Cl Nc1cc([N+](=O)[O-])ccc1C(=O)NCC(CNC(C1CC12CCC2)=O)CO c1(OC)cc(C(C)NC(N2CCN(Cc3coc(C)c3)CC2)=O)ccn1 CC(C)CCC(=O)NC1CC(C)N(C(C2CC3C=CC2C3)=O)C1 C1(CNC(C(CC)=CC)=O)CCC(C)(C)CN1C(c1ncccc1N)=O C1(CNC(C(C)c2ccco2)=O)COCCN(C(=O)C=Cc2cnc[nH]2)C1 C1(NC(CCc2cc(C)on2)=O)CN(C(c2cc3c(s2)CCC3)=O)C2(CCC2)C1 c1(C(=O)NC(C2N(C(COCCC#C)=O)CCCC2)C)ccc(C)cc1Cl CCC(F)(F)C(C)(C)C(=O)N1CC(CCNC(C2CCOC(=O)CC2)=O)C(C)C1 N(C1CCCOc2ccccc21)C(=O)OC(CN1CCC(C2CC(C(C)(C)C)C2)C1)=O n1(CCCC)nccc1C(N1CC(CO)(NC(C2CC2C)=O)C1)=O N1(C(c2ccc(CC)cc2N)=O)CC2CCN(C(=O)C(N3CCOCC3)C)C2C1 c1(NC(CC(C)C)CO)ccc(C(F)(F)F)cc1S(=O)(=O)NCCC1CCOC1 c1(OC)ncnc(C(N2CC(NC(=O)CCn3c(C)ccc3C)C(C)C2)=O)c1F c1(C(N2CC(OC)C(NC(C3CCCC3C)=O)CC2)=O)ccc2c(c1)CCCO2 C1(CC(=O)NC(C)CNC(=O)CC(c2cccc(F)c2)C)CCCS(=O)(=O)C1 c1(CC)onc(C)c1C(=O)NC1CC(n2cc(C3CC(F)(F)C3)nn2)C1 N1(C(C(CC2CN(C(C=CC(CC)C)=O)C2)F)=O)CC(C(=O)NC)CC(C)C1 C1(NC(c2cnn(-c3ncc(Cl)cn3)c2)=O)CC2CCC1(NC(C1CCC1)=O)C2 C=C(Cl)CC(C(=O)NCCOCCC)NC(c1ccsc1Cl)=O C1(CNC(c2c(CC)cc[nH]2)=O)CCC2CN(C(c3nccnc3N)=O)CC12 N1(C(C)=O)CCC(C)(C(=O)NC(C)CCCNC(c2ccncc2N)=O)C1 Cc1cn(C)nc1C(=O)NC(CNC(=O)CCC1CCC(=O)N1)CO C12(NC(c3oc(C)c(C(C)C)n3)=O)CCCC1CN(C(=O)CN1CCCCC1)C2 CCCCC(CNC(C1(C(C)C)CC1)=O)NC(=O)C(F)CC N1(C(c2nc(C)nc(O)c2)=O)CCC(F)(F)C(CNC(=O)C2=C(Cl)CCC2)C1 c1(C(=O)NCC2=CCN(C(C(C(=O)OC)(C)F)=O)CC2)cccc(Cl)c1[N+](=O)[O-] c1(C(=O)NCC2CCN(C(CCS(C)=O)=O)C23CCC3)cc(Cl)c(F)c(Cl)c1 C1(NC(=O)COC(F)F)CCN(C(=O)C(c2cc(F)cc(Cl)c2)=O)CC1O c1(C(=O)NCC)cc(F)ccc1NC(=O)Cc1cn(-c2ccc(C)cc2)nn1 c1(CC(=O)N(C2CCN(C(=O)C=CC(C)C)C2)CC)ccc(F)c(OC)c1 c1(C(N2CC(O)CC(NC(c3ccc(C#N)[nH]3)=O)C2)=O)cccc2nn[nH]c12 c1(CNC(N2CC(C(C)C)OCCC2)=O)cc(F)cc2c1CCC2 C1(C(CC)NCc2sccc2S(N)(=O)=O)Cc2ccccc2C1 N1(C(COCC(=O)NC)=O)CC(CN(C(=O)CC(C)C(=O)OC)C)C2(CC2)C1 C#CC1CCC(NC(=O)C(=O)NCCc2cn(C)nn2)C1 C1(NC(C2CC2Br)=O)CCC2CC1CN2C(c1cccc2c[nH]nc12)=O c1(OCC)c(F)c(-c2nc(C(C)C)no2)cc(F)c1F.N12CCC(CC1)C2=O N1(C(C2CC(CC(=O)O)OCC2)=O)CCC2CCCC12 C(=O)(C1Cc2ccccc21)N1CCC(CC)C1C(=O)N(C)Cc1nc(C)no1 c1(NCC2CN(S(C)(=O)=O)C2)ccc2ccc(Cl)c(Cl)c2n1 c1(C(N2CC(C(N3CCC34CCCCC4)=O)C(F)(F)C2)=O)c[nH]c2ccccc12 C=CC1CN(C(c2cncc(C3CC3)c2)=O)CC1NC(C1CC(CC)C1)=O C1(NC(CCOC)=O)CCCC12CN(C(c1cccc(N3CCNC3=O)c1)=O)C2 COn1cnc(C)c1C(=O)NCC(O)CC(=O)NC1COCCOC1 C(C)(CCCCn1cc(-c2sc(CO)cc2C)nn1)NC(C(C1CCCCC1)C)=O c1(CNC(CSc2c(OC)c(OC)ncn2)=O)ccc(F)c2c1CCC2 Cc1cccc(NC(=O)NCC2CCN2C(C)Cc2ccccc2F)c1 N1(C(C(C)N2CCC2)=O)CCCC2(CCN(C(C34CCC3CC4)=O)CC2)C1 C1(N(C(=O)C(C2CCC(=O)CC2)F)C)CN(C(c2cnc(O)s2)=O)CC12CC2 CCC(C)C(=O)C(=O)N1CC(C(=O)Nc2ccc(COC)nc2)OC(C)C1 c1(SC)cc(C(N2CCCC(C(C)NC(C3(O)CCOCC3)=O)C2)=O)ccc1F CN1C(=O)NCC12CN(C(=O)COC1CCN(C(=O)CCC3CC3)C1)C2 CC(C)C1=NOC(SC(C2CCC(n3cc(C4C(C)CCC4C)nn3)CC2)=O)C1 C(c1ccc(F)cc1)=C(C)C(=O)NCC1CC1NC(=O)Cn1cc(CO)nn1 Cc1cc2c(C(N3CCC(CNC(=O)CN(C)CC4CC4)CC3)=O)nccn2n1 C(CCCCC(=O)NC1(C)CCN(C(=O)C(C)(C)C(C)C)C1)=CC C1(C(N2CCN(C(c3c(CC)scc3)=O)CC2CO)=O)CCC(S(C)(=O)=O)CC1 S(=O)(=O)(c1cc([N+](=O)[O-])ccc1Cl)N1CC(CC(C)C)NC(=O)C1 c1(C(=O)NC2(C)CCN(C(CC(CC)C(F)F)=O)C2)csc2c1C(C)(C)CCC2 C(=O)(CC(C)(C)C=C)N(CC(c1ccccc1)NC(C(C)OCCC#C)=O)CC N1(C(=O)CN2CSCC2=O)CCSCC1CC(c1ccccc1)=O Cc1ccc2c(c1)CC(C(N1CCN(C(c3cn4c(n3)CCC4)=O)C(C)C1)=O)S2 N1(C(c2cc(OC)nc(C)c2)=O)CC(C)CN(C(C2(CN(C)C)CC2)=O)CC1C C1(C(=O)NCC(C)(C2CCC2)NC(c2ncccn2)=O)CCCOC1 c1(C(=O)NC2(CNC(Cc3c(C)nc[nH]3)=O)CCC2)cnnc2ccccc12 c1(C(C(=O)NCCC)N(CC(=O)N(C)CCOC)C)cnc(C)c(NC)c1 CCC(C)C(O)C(C)C(=O)NC(CC(N1CCC=C(F)C1)=O)C1CC1 c1(C(N2C3CN(C(COCCSC)=O)C(C3)C2)=O)ccsc1S(N)(=O)=O O=C(CCCn1cccn1)NCC1CC(O)(CNC(C2CCOC2F)=O)C1 C(=O)(C(O)CCNC(=O)CN1CCOC(C)C1)NCCCC(=O)OC C(=O)(CCC(CF)CF)N1C(C(=O)NC2C(O)C3CCOC23)CSCC1 CC1CCC(C(=O)NC2(CCC(=O)N(C)CCN(C)C)CCCC2)O1 c1(C(=O)NC(C)CCNC(c2n[nH]cc2[N+](=O)[O-])=O)cc2nccc(Cl)c2s1 C1(NC(c2c(CC)nn[nH]2)=O)CC12CCN(C(=O)COc1ccc(F)cc1)CC2 N1(C(c2cccc(C)c2)=O)C(C)C2CC1C2NC(=O)C(O)CN1CCCC1 c1(CN2CCC(NC(c3ccnnc3)=O)C(O)C2)ccc(Cl)c([N+](=O)[O-])c1 N#CC1C2CC2CN1C(c1cccc(-c2ccco2)c1)=O c1(OC)nccc(C(=O)NC2CCCN(C(=O)OC(C)(C)C)C2)c1Br C1(C(=O)NC2C(C)CCC2C)CCC2(CC2)N1C(C1CCC(N(C)C)CC1)=O c1(NC(C(=O)NCC(C)S(C)(=N)=O)=O)ccc(Cl)c(S(N)(=O)=O)c1 C12CCC(C)(CC1)C(=O)N2.C1(COCC)CCN(C(=O)NC(C)C)CC1 C(=O)(C(CNC(C1Cc2cccnc2C1)=O)C(C)(C)C)NC(c1nc[nH]n1)CC CC12CCCC(C(=O)NCCC3(O)CCN(C(C4(F)CC=CC4)=O)C3)(CO1)C2 C=CC1(C(=O)NOCC(O)CO)CN(C(=O)CC2CCCC3CC23)C1 n1(C(CC)CC)nc(C2CC2C(C)C)nc1C1CC1C1CC1 CN1CCCCC1C(=O)NC(C)(C)CN(C)C(C1CCN(C2CCCCC2)C1)=O C1(C(N2CCC(C(=O)NC3(CC(N)=O)CC3)(OC)C2)=O)(CC)CC(C)(C)C1 C(CC(=O)NC(c1cccs1)C)(C(F)(F)F)NC(C(CCC)NC(N)=O)=O CCC(O)CC(=O)NC1C=CCC(C(=O)NCC2CCCC2)C1 C1(NC(c2ccc(-n3cncn3)c(F)c2)=O)CN(C(c2cocn2)=O)CCC1CO N1(C(C2(OC)CCOC2)=O)CC(C)CN(C(=O)COC(C)C)CC1C c1(C(=O)NCC2(C)C(NC(CC=CC=C)=O)CCC2)cccc2occc12 CN1CCC(C(=O)NCC2CN(C(c3c(F)cccc3Cl)=O)CCN2C)CC1=O C1(NC(C=C(C)I)=O)CC(CNC(C2CC2(F)F)=O)C1 CCC(C)(CC(c1nnnn1C)NCCOCCOCc1ccc(C)cc1)OC c1(C(=O)NCCC2(C)CCN(C(CCn3c(C)ncc3)=O)C2)cc(N)c(F)cn1 Cc1cc(C(=O)NC2CC(CNC(c3cc[nH]n3)=O)C2(C)C)ccc1Br C=CCC(CNC(=O)C(CC)=CCCC)C(=O)N1CCN(C(C)=O)C(C)C1 N1(C(=O)CC2CCC3CC23)CC(F)(c2cn(Cc3nc(C(=O)O)co3)nn2)C1 C(=O)(CCC(F)(F)F)N(CCC(N1CCC(C(C)C)C1)=O)C C1(CNC(C(CC=C)(F)F)=O)CCN(C(c2cc(Cl)ncc2N)=O)CC1(F)F C1(C2(O)CCN(C(c3[nH]ccc3C3CC3)=O)CC2)(NC(=O)CC2CSC2)CC1 c1(C(N(CC(C)CNC(C2CCC2C(C)(C)C)=O)C)=O)cc(Cl)cc([N+](=O)[O-])c1 CC(C)C(C(=O)N1CCC(c2ccon2)C1)C(C)C.c12cncc(c1)C(=O)N2 c1(C(=O)NCCCN(C(=O)C(C)(F)CC)CC)cccc(-c2ccccc2)c1 C1(NC(C(=O)N(C(C2CCCO2)C)CC)=O)CC2CCC1C2 Cc1csnc1C(=O)NC(C)CCCNC(=O)C(C)NC(C)C(C)C C1(NC(C=C)=O)CCN(C(C)=O)C1(C)C.C1CC1 C(CCF)(C(=O)N1CC(N2CCCC2)C1)NC(CC(C)n1cccn1)=O C(CC)(CC)(CCNC(=O)C(C)SCC)NC(C=CC)=O C=CC(C)(C)CC(=O)NCC(C(=O)NCC12CCCC1CCC2)N(C)C N1(C(C(C)Oc2ccccc2)=O)CC2(NC(=O)C(C)C3(O)CCC3)CCC1C2 Cc1n[nH]c(C)c1CCC(N1CC(NC(=O)C(F)(F)c2cnccn2)CC1C)=O c1(SCC(C)Oc2ccccc2)ccc(N2CCNS2(=O)=O)cc1 C1(NC(C(CC)SC)=O)CC2(C1)CC(CNC(c1ccnn(C)c1=O)=O)C2 N1(C(c2c(C(C)C)occ2)=O)CC2CC2(C(=O)N(C2CC2)C2CC2)C1 N1(C(c2oc(C)c(Br)c2)=O)CCCC(NC(=O)C(O)C(F)F)C1C N1(C(C2C(CC)CN(C(=O)C(=O)N(C)C)C2)=O)C(CO)CC2CCCC12 Cc1cc(C(N2CCCC(Cn3cncn3)C2)=O)nnc1O C(C(CC(C)C)C(=O)N1CCN(C(c2snnc2C)=O)CC1CF)OC CCCCCC(C)(C)C(=O)NCC(C1CCOC1)NC(=O)C(C)(C)c1cc[nH]n1 c1(CC(=O)NCC#CCNC(C2C(=C)C2)=O)cccc(N)c1 C1(NC(C(CCC)C)=O)CCC2(CCN(C(=O)C3=CCCCC3C)C2)C1 C(C(C)C(C)C(=O)NCC1(CCNC(=O)Cc2c(C)ncnc2C)CC1)OC C1(C(=O)NCc2cc(C)c(-n3ccnc3)cc2)CC=CC(N=[N+]=[N-])C1 CCCC(C)C(C(=O)Nc1ccccc1Br)N(CCCF)Cc1cc(Cl)cc(Cl)c1 C(CCCCC(=O)NCC(C)CN(C)C(C1CC(CCO)C1)=O)SC C1(C(=O)NCC(CC)NC(c2ccc(N(C)CC)cc2)=O)CCCN(C(C)=O)C1 c1(C(C)NC(=O)CSCCNC(=O)C(C)c2cccs2)cnccn1 C1(NC(C2CCC(C)(F)CC2)=O)CC12CCN(C(c1cc(C(F)F)cs1)=O)CC2 N#Cc1cc([N+](=O)[O-])cc(Br)c1NC(C1CC(F)(F)CN1C(=O)C1=COCC1)=O CCCCC(CN(C(=O)CC1CC(F)CN1C(c1cc(C)cs1)=O)C)CC c1(CC(C(=O)OCC)NC(C2CC(C#N)C2)=O)ccc(N)cc1 C(=O)(C1Cc2ccccc21)NC1CC(NC(Cc2cn(CC)nn2)=O)C(O)C1 N1(C(CC23C(CN(C(c4c(C)ncs4)=O)C2)CC3)=O)CCN(C)C2(CC2)C1 C1(N(C(=O)CC2(C)CCCO2)C)CCC(CNC(=O)COC2CCCC2)CC1 c1(CCC(=O)NCC2(COC)CCC2)cc(C(=O)NCC2CCCO2)n[nH]1.CC c1(C(=O)NCC(CC)NC(=O)CN2CC3CC3C2)ccc(F)c(Cl)c1N C1(CC(=O)NC(CC2CN(C(c3cc(C)ns3)=O)C2)C)CC2CCC(C1)C2 C(=O)(C(O)CC(N)=O)NC1C(C(=O)NC(CC=C)C(=O)OCC)OCC1 C12(C(=O)NC3C(CNC(CSCCC)=O)CC3)CC(CC)(CO1)C2 c1(C(C)(C)C)n[nH]cc1C(=O)NCCOC1CN(C(c2n[nH]c(C(F)F)n2)=O)C1 C1(CNC(c2c(CC)onc2)=O)C(C)CCN1C(C1CC(OC(F)(F)F)C1)=O c1(CCCC(=O)NCC2CC(NC(COCCC)=O)C2)ccccc1Cl Cc1cc(=NC2CCN(C(=O)C=Cc3ccccc3F)C2)c([N+](=O)[O-])c(C)[nH]1 N1(C(c2cocc2Br)C(=O)NCCCF)CCC(C2=NOCC2)C1 c1(OC)ccccc1N(C(=O)C#CCNC(=O)CC1CCC(C#N)C1)C N1(C(c2n(C=C)ncc2)=O)CCC(C2CC2)C1C(=O)NOCCC(C)O C(CC(F)=C(F)F)NC(c1n(CC(=C)C)nnn1)c1ccc(I)s1 CCC(C)C(C(=O)N1CC2CC1(C(=O)NC1(CC3CC3)CC1)C2)OC c1(OC)cc(C(=O)NCC(F)CNC(C2(C3CC3)CC2(F)F)=O)ccc1[N+](=O)[O-] c1(C(N2CCCC(CN=[N+]=[N-])C2)C(=O)NCC=C)cc(C(=O)OC)c(C)n1C C1(C(=O)NCCC(C)c2cn[nH]c2)CN(C(=O)CN(C)C)CC1CO N1(C(Cc2cn(C)nn2)=O)CCC2(CCC2)C(NC(C2CCC2(C)C)=O)C1 C1(C)(C(=O)NCCN(C(CC2CC(OC)C2)=O)CC2CC2)CCCNC1=O CCCCC(O)CC(=O)NC(C)(CNC(c1cnc(C)o1)=O)CC c1(C(=O)NCC(CN(C(=O)C=Cc2cnc[nH]2)C)O)cc(Cl)nnc1O c1(OC)cccc2c(N3CCC4(CNC(=O)C(C)CF)CCCCC34)ncnc12 c1(CC(=O)NCC(C(C)(C)C)NC(CC=C=C)=O)c[nH]c2ncccc12 O(N(C)C(=O)CC(CN(C)C)CC)C(C(=O)OC)(C)CO.CC(=O)N C(=O)(C1CSc2ccccc21)NCCCNC(c1ccc(C#C)cc1F)=O CC(CCCNC(c1scnc1C(F)F)=O)NC(=O)CC1CCCC1C Cc1noc(CCCC(=O)N2CCC(CN(C3CCC3)CC(C)C)C2)n1 c1(C(=O)NC(CN(C(c2c(COC)noc2)=O)C)C)sc(-c2nc[nH]n2)nc1C C=CCC(CC(=O)NC(C=C)CO)NC(c1ccc(C)nn1)=O c1(C(=O)NC2(CNC(C3CN(C)C(=O)C3)=O)CCC2)cnn2cc[nH]c12 C(=O)(C1=CCCCCC1)NCC(C(=O)N(C)Cc1nc(C)sc1)CC1CC1 C1(NC(C2(OCC)CCCC2)=O)CN(C(=O)CCCF)C2(CCCOC2)C1 c1(C(N2CC(F)(CNC(c3[nH]cc(C)c(=O)c3)=O)C2)=O)cc(F)c(F)cc1O C1(C(=O)NC(CNC(c2cc(OCC)ncc2)=O)CC)CC(C2CCCCC2)C1 c1(C2C(NS(CCSCC)(=O)=O)CC2)ccc(Cl)cc1F c1(C(=O)NCc2cc(OCC)n[nH]2)n[nH]c2c1CN(C(=O)CSC(C)C)C2 CCC(CC(=O)N1CC2CC1C2NC(=O)C(C)Cc1cnc[nH]1)CC(C)C c1(C(N2CCC(CNC(=O)OC(C)(C)C)C2)=O)ccc2c(c1)NC(C)CC(=O)N2 C1(CC(=O)NC23CCC(OC)C2C3)CCN(C(c2ccc(CO)nc2)=O)C(C)C1 c1(C(=O)NCC(C)NC(=O)CNC(=O)CC(F)(F)F)cc([N+](=O)[O-])ccc1Cl CC1CC(N)CCN1Cc1ccc(F)cc1Br N1(C(C(C2CCCCC2)NC(CCC(CC)OC)=O)=O)CCOCC(C)(O)C1 C(CCC(O)C(=O)N=c1ccn(C)[nH]1)NC(C(CC)=CCCC)=O c1(CC(C(=O)O)N(CCN=O)CCNc2ncnc(C)c2C)c[nH]c2nccc-2c1 N1(C(CN(C(C)=O)C)=O)CCC(C(=O)NC2CC(O)C2)C1C(C)C N1(C(C2C(c3c(C)ccs3)C2)=O)CC(NC(=O)CCOCC(C)(C)C)C2(CC2)C1 CCC(CC(=O)NC1CN(C(=O)COCC(C)C)C(C)(C)C1)C(F)F N1(C(CCOC)=O)CCCCC12CN(C(=O)C(N1CCSCC1)C)C2 C(=O)(NNC(=O)CN1CCN(c2ccc(F)cc2Br)CC1)c1cc(OC)ncc1 Cc1nc(C)c(CC(=O)NCCCN(C(=O)C(O)C2CCCC2)C(C)C)s1 C=CCCCCC(=O)N1CCCC(CO)(NC(=O)C(C2CCCC2)OC)C1 C1(C(=O)NCCOCC(N)=O)CCN(C(=O)C(F)CC2CC2)C12CCC2 C1(C(=O)NCC2N(C(c3ccc(C)o3)=O)CC2)CCCCC1c1nc(S)n[nH]1 C1(NC2(c3nnnn3CCC)C(CCCC)CCC2)CCOC2(CCOCC2)C1 N1(C(C2CC3(C2)OCCO3)C(=O)NCCCSC)CC(F)(F)C2(CCCC2)C1 C1(NC(c2nc3ncccn3n2)=O)CCCC2CN(C(=O)C=C3CCC3)CC12 c1(C(N2CCC=C(Br)C2)C(=O)NCC(=C)C)cccc(C(C)(C)C)n1 CN1CC(O)CC1(C)C(=O)NCC1CN(C(=O)C=C2CCC(C)(C)CC2)C1 N1(C2CCN(C(c3ccccc3-c3c(O)cccc3O)=O)C2)CCC2(CCCO2)C1 C1(CNC(C2C(OCC)C2)=O)CC2(CC2)CN1C(=O)COc1cccc(Cl)c1 c1(C(N2CCCC(C)(CNC(=O)CSCC(N)=O)C2)=O)ncn2cc(Cl)ccc12 C(=O)(C(F)(F)C(C)(C)O)NCC(CC)NC(c1ccccc1-n1cccc1)=O c1(C(N(C2CCC(NC(=O)C(O)CC(C)(C)C)C2)C)=O)ccc(F)c2occc12 N1(C(C=CCOC)=O)CCC2C(NC(c3cccc(C4CC4)n3)=O)C2CC1 CC(C)C(O)C(C)C(=O)NC1C2CC3C(C2)C13C(=O)NCC(C)(C)C(C)(C)C C1(C(=O)NCC)(OC(CC2(CCC)CCCNC2)=O)CCS(=O)(=O)CC1 c1(C(=O)OC)cc(C(N2CCOC(CSC3CCCCC3)C2)=O)cc(C2CC2)c1 C#CCC(C)(C)C(=O)NC1CCC(CCNC(=O)C(F)F)C1 C1(NC(CNC(C)=O)=O)CCC12CCN(C(=O)C(c1ccn(C)n1)C)CC2 N1(C(CCNC(CC(C)C)=O)=O)CC(NC(C2(C(F)F)CC2)=O)CC(C)(C)C1 CC(N=c1cc[nH]cc1S(=O)(=O)NC1CC=CC1)C(F)F n1(CC)ccnc1C=CC(=O)NC(C)(CNC(=O)CC(C)OC)C1CCC1 N1(C(CC(C)C(F)F)=O)CCCC2(CCN(C(c3nnc(C4CC4)s3)=O)C2)C1 C(=O)(CCCCC#N)NC(C(C)NC(c1noc(C)c1Br)=O)C(C)C N1(C(CCC=CC(C)C)=O)CC2CC(NC(C3CC(=O)NC3(C)C)=O)CC1C2 C1(N(C(=O)CCSC(F)(F)F)CCOC)CCN(C(C2CCC(NC)C2)=O)CC1 C(CCCCCCC(=O)N1C2CCC1CC(CNC(=O)CCS(C)=O)C2)SC C(=O)(C(O)CC(C)(C)C)NC(CCN(C(Cc1nc(C)oc1)=O)C)C(C)(C)C CCCCC(CN=c1[nH]cnc2ccccc12)NC(=O)C(F)(F)C1CC1 C(=O)(CC1=CCOCC1)NC1(C(=O)NC2CCC(C#C)C2)CC(F)(F)C1 C1(C(N(C2CN(C(C3CC(=O)NC(=O)C3)=O)CC2O)C)=O)C(C)(C)OC1(C)C N1(C(C(CNC(c2c(OC)nsc2)=O)CC2CC2)=O)CCSCC(C)C1 Cc1cc(C(=O)NC2CCCC2(C)CN(C(=O)CC2(C3CC3)CC2)C)sc1Cl C=C1CC2(C1)CC(C(=O)NCC1(C(N)=O)CN(C(c3ccnc(C)n3)=O)C1)C2 C1(C)(CCNC(CCN(C(=O)CCC2(C)N=N2)C(C)C)=O)CC1(F)F c1(NC23CCC(NC(C4(COC)COC4)=O)(CC2)C3)ncc([N+](=O)[O-])cc1Br c1(OC)cccc(Cl)c1CC(N1CCC(N(C)CCO)C1)=O.N12CCNC(C1)C2=O C1(NC(=O)C=C2CCCCC2)CCN(C(=O)CCCN2CCOC2=O)CC1O c1(CC(=O)OCC(c2cccc(Br)c2)C)ccc(C(F)(F)F)nc1 Cc1cc(N2CC(C(N3CCC3NC(C3(C#N)CCC3)=O)=O)CC2=O)cc(F)c1 N1(C(Cc2cccc(N)c2)=O)CCC2(CCCCC2NC(c2c[nH]nc2F)=O)C1 C(=O)(CC(C)(C)CNC(=O)C(F)C(F)(F)F)NCC(C(C)O)C c1(C(N2CCC(C)(NC(c3n(C)cnc3)=O)C2)=O)ccc2c(c1)CCNC2=O N1(C(c2cc(C)no2)=O)CCC(CC(=O)NCC2CCN(C(C)C)C2)C1(C)C C1(CNC(C(C2CCCC2)NC(c2n(C=C)ncc2)=O)=O)CCCCC1(C)C c1(OCC(N)=O)ccc(C(N2CCN(C(c3c[nH]nc3Br)=O)CC2)=O)cc1 c1(C(=O)NCCC(C)NC(C2(CC)CCOC2)=O)cccc2ccoc12 C1(NC(C(COC)C)=O)(CNC(=O)CCn2c(C)ccc2C)CCOCC1 c1(C(=O)Nc2ncc(C(=O)OC)s2)cnc(N)cn1 C(=O)(C(C)CCC(C)(C)C)N(CCC(=O)NCCNC(C(C)C)=O)CC1CC1 c1(C(=O)NCC2CC2NC(C2CCCS2)=O)ccc(OC(F)(F)F)nc1 C1(NC(c2coc(-c3ccccc3)n2)=O)CN(C(C2CC3(CC3)CO2)=O)CC1O c1(C(=O)NC2CCN(C(C3(n4ccnn4)CC3)=O)C2)cncc(OC(F)(F)F)c1 C1(CC=C)(C(=O)N(C)CCc2ccccn2)CCN(C(c2ncncc2N)=O)C1 C(=O)(C1=CCN(C(C2CCCC(=O)N2)=O)CC1)NC1CN(C)C(=O)C1 c1(CC)noc(C)c1C(=O)NC(C1CCOC1)CNC(c1cnc(C(C)C)s1)=O Cc1nc(N2CCCC2)ncc1C(=O)NC(CNC(=O)CN1CCC1C)C1CC1 C(C1c2ccccc2CCN1C(c1c(C)nsc1C)=O)NC(C(C(CC)C)C)=O c1(OCC)cnc(F)c(CNC2CCN(C(=O)OC(C)(C)C)CC2C(=O)O)c1 c12ccc(F)nc1S2.CC(CC(F)(F)F)NCCO.c12nnc(C(F)(F)F)n1C2 c1(C(N2C(CNC(C(CCSC)O)=O)CC(O)C2)=O)cc(P(C)(C)=O)cs1 CCCC(CC)CC(=O)NCC1(O)CCN(C(=O)CC(c2cccc(F)c2)C)C1 c1(SC)nc(C(F)F)cc(=NC(C)CC(C)NC(=O)Cn2ccnn2)[nH]1 C1(C(F)(F)F)(C(=O)NCCC2CC(NC(c3cc(OC)ns3)=O)C2)CC=CCO1 C1(C2CCN(C(c3ccsc3C(F)F)=O)CC2)(NC(c2ccsn2)=O)CC1 N1(C(CN(C2CC2)CC)=O)CCC(NC(=O)C(c2cccs2)SC)C1C1CC1 CCCC(O)CC(=O)NC(C1(O)CN(C(=O)Cc2cccc(Cl)c2Cl)C1)C N1(c2n(CCCC=C)ccn2)CCc2sc(-c3cc(OC)c4nccn4c3)nc2C1 Cc1ccnc2c(C(=O)NC34CCCC3CN(C(c3sccc3F)=O)C4)cnn12 C(CCCCC(=O)NC(C1CCCC1)CNC(=O)C(C)(F)F)OC N1(C(=O)NC(C)CC2CC2)CCS(=O)CC1c1cnn(C)c1 c1(C(C)C)ccc(N)c(C(N2CC(NC(=O)C(O)CCN(C)C)C(O)C2)=O)c1 c1(C(=O)NC23CC(COCCOC)(C2)C3)[nH]nc2ncccc12 C(CCC(C)C)(C(=O)N(C1CC1)CC1CCCCC1C)NC(c1c(C)scn1)=O O=C1CCc2cc(C(N3CC(O)(CNC(=O)C4CC4)C3)=O)ccc2N1 N1(C(C(N2C(C)CCC2C)C)=O)C2CCC1CN(C(C1CCCOC1)=O)CC2 CC1CCN(C(=O)CN2CCC(C(F)(F)F)CC2)CCN1C(C12CC(F)(C1)C2)=O N1(C(C2C(OC)CCCC2)=O)CCN(C(=O)CCCCC2CC2)C2COCC12 C1(C(N2C3C(NC(=O)CN4CCCCC4=O)C(C3)C2)=O)CCCCNC1=O n1(CC(=O)N(CC(CO)(CO)NC(C(C)=C2CC2)=O)C)nc(C)c([N+](=O)[O-])c1C CC1CN(C(c2ccsn2)=O)CC(C)C1NC(c1c[nH]cc(Br)c1=N)=O C1(C(N)=O)CCCCC1CNC(=O)C(N1CCC(Nc2ccccn2)CC1)=O Cc1ccc(C)c(C(N2CCC(=CCNC(C3CCCC3C)=O)CC2)=O)n1 C1(C(=O)NC2CCCC(C#C)C2)CC2(CCN(C(c3cn(CC)nc3C)=O)C2)C1 C1(CN(C(=O)NC(c2nc(C)oc2)C)C)CCCN(C)C1 O=C(CCC(=O)N1CCC(CNC(c2cnoc2C2CC2)=O)C1)c1ccncc1 c1(NC(NC(C23CC(C2)C3)=O)=S)nc(Cl)ccc1O c1(C(=O)NC2CN(C(C(OC)OC)=O)CC2SC)cnc2ccc(F)cn12 C=CCC(CNC(=O)C(C)CC(N)=O)C(=O)NC1CC(O)C1 C1(OC)CC(C)CN(C(C2CC(F)(F)CN2C(=O)CN2CC(C)(C)C2)=O)C1 c1(C(N2C3CN(Cc4c(F)cccc4Cl)CC23)=O)ccc2c(c1)CNC2 C(=O)(N=c1cc(C#N)[nH][nH]1)C1(O)CCN(C(=O)C(O)C(C)(C)C)CC1.CCC=O C12CCC(C1)NC(=O)CCC2.C=C1C(C(=O)OC)C1C(=O)NC(c1cccs1)=O N1(C(c2ncc(OC(C)C)nc2)=O)C2CCCC1CN(C(C1CC1(F)Cl)=O)C2 c1(N(C)C)cnc(Cl)c(C(N2CCC2C(=O)Nc2ccc(Br)cc2F)=O)c1 N1(C(c2c(C)cncc2)=O)CC(NC(c2onc(C)c2C)=O)CC(C)(C)C1 C1(C)(CNC(Cc2cc(C)ns2)=O)CCCN1C(=O)CC(C1CCC1)C1CCC1 C1(NC(CC2C(C)(C)C2(C)C)=O)CCC12CCCN(C(=O)C=CC1CC1)C2 C(CNC(=O)Cc1ccnc(C(=O)N(C)C)c1)(CC(=O)N1CCC1C(N)=O)OC C12CN(C3(CCC3)C1)C2=O.C(=O)(CC(F)(F)F)C(CCc1onc(C(C)C)n1)=O C1(CNC(C(C)OCCC(C)C)=O)C(C)CCCN1C(C1SCCCS1)=O C1(C(=O)NC(C#C)C(C)OC)CC2CC2N1C(=O)CN1CCCNC1=O Cc1ccc(C)c(C(N2CC3CC3(CNC(=O)CSC(C)(C)C)C2)=O)n1 C=CC(C)CC(=O)NCCCCNC(=O)CCC1CCC1 C#CC1CN(C(c2ccn3nnnc3c2)=O)CCN1C(=O)C(F)=CCC Cc1nc(C=CC(N2CCC3(NC(=O)CSCC(F)(F)F)CC3C2)=O)[nH]c1C c1(C(N2C(C(C)NC(Cc3c(C)ccs3)=O)CCC2)=O)cc(F)n(C)n1 N1(Cc2cnc(C)nc2)CCc2c(C(N3CCC(O)C(C)(CO)C3)=O)csc2C1 C1(n2cc(CSC)nn2)CC2CCC1(NC(c1ncccc1Br)=O)C2 N1(C(C=Cc2cn(C)nc2)=O)CCC2(CC1)CN(C(c1cnco1)=O)C2 C1(C(N2CC(C)(NC(c3ccc(F)c(Cl)c3)=O)C2)=O)CCCCC12CC2(F)F c1(N(C)C)ccc(N)c(C(N2CC(CCNC(=O)CCC3CCOC3)C2)=O)c1 CCCC(CNC(=O)CC1CCC1)C(=O)Nc1csnc1NC Cc1c(C(N2CCCC(NC(=O)C(O)CC(F)(F)F)CC2)=O)[nH]c2ccccc12 c1(C(N2CC(CNC(CC3CCC(C)C3)=O)C2)=O)cc2nc(Cl)ccc2o1 C1(N(C)C(c2ccc(C(F)F)o2)=O)CCN(C(C2CC2(C)C)=O)CC1 C1(NC(C2C(C(=O)OC)C=C2)=O)CCCC(C2CC2)C1.C12(CC1)C(=O)NC2 CNS(=O)(=O)NCC(N1CCCC1C(C)(C)CNC(C1(C)CCOC1)=O)=O C1(C(=O)NCC2C(NC(c3c(CC)ocn3)=O)CC2)C2(CCC2)C12CCC2 c1(C(=O)NC2CCC(NC(c3cc(C#N)no3)=O)CC2)cncc(Cl)c1Cl c1(C(N2CCC(N(C(=O)C(C)SC)CC)C2)=O)ccc2c(Cl)nccc2c1 C1(CC(=O)NCCCSC2CC2)CCCN(C(c2cncc(CO)c2)=O)CC1 c1(C(=O)NC2C(CNC(CCOCCOC)=O)CCC2)cccc2c1CCN2 CC1(C)COC(CC(N2CCCC2CNC(=O)CC(=O)OC(C)(C)C)=O)CO1 Cc1ccc(C(N2CC(CC(C)NC(=O)Cn3cc[n+](C)c3)C2)=O)c([N+](=O)[O-])c1 c1(CNc2ccoc2Cl)ccnc(O)c1Br.C12C3CC1N(C3C)N2C(C)C Cc1ncsc1CN(C(C1CC2CC2C1)C(=O)NC1CC1)C c1(C(=O)NC2CCCN(C(c3nc(Br)c[nH]3)=O)C2)noc2ccc(Cl)cc12 c1(C(=O)NCC2(NC(CCC(C)(C)F)=O)CC2)oc2ccccc2c1CO.CC#N c1(C2C(C(N3CCC(N(CCC#C)C(C)=O)C3)=O)C2)cc(Cl)cc(Cl)c1Cl C1(CNC(CC2(C)CC2(Cl)Cl)=O)CC2(CC2)CN1C(=O)Cc1ccsn1 C1(CC)CCOCCN1C(=O)CC1(NC(=O)CCC(C)(C)c2ccccc2)CC1 Cn1cc(C(=O)NCC2CCCC2NC(c2cnnc(O)c2)=O)c(C2CCC2)n1 Cc1ncc(N)cc1C(N1CCC(NC(c2cnn(C)c2C)=O)C(C)C1)=O N#Cc1csc(C(=O)NCC2CN(C(c3occc3Cl)=O)C2)c1 C12(C(N3CCC(C(C)NC(C(C)N(C)C)=O)CC3)=O)CCOC(C)(C1)C2 Cc1cn(C)nc1CCCn1cc(C(=O)NC(c2csc(O)n2)=O)nn1 Cc1nccc(C(=O)NC(CNC(C2(C(C)C)CCC2)=O)C(C)C)n1 CCCCCCC(F)C(=O)NCCCCNC(=O)C(CC)OCCOCCSC C1(NC(C2N(C(C)(C)C)CC2)=O)CC2CN(C(c3sccc3Cl)=O)CC12 N1(C(C2C(C)(C(F)F)C2)=O)CC(N(C)C)C(CNC(=O)Cc2cncs2)C1 N1(C(C=CC(C)(C)SC)=O)CCCN(C(=O)Cc2cn(C)nn2)CC1 c1(C(N(CC(C)NC(C2(CC(F)F)CC2)=O)C)=O)cscc1Br N1(C(C(C)=CC)=O)CCCCC2(CCN(C(=O)CCc3ccc(C)o3)C2)C1 c1(C(=O)NCC(CNC(C2(SCC)CC2)=O)(C)C)c(O)ccc(C)c1C N1(C(C2CCCN(C(c3c(C)con3)=O)CC2)=O)CC2CC(C1)C2(C)C N1(C(c2c(C)cn(C(C)C)c2)=O)CCC(C2(NC(=O)C=CCF)CC2)CC1 O=S(=O)(c1ccc(NCCOCC2CC2)c(Br)c1)NC1(Cl)CC1(F)F C1(N(C(=O)CC=CC(C)(C)C)C)CN(C(=O)C=CC(C2CCCC2)=O)CC1F Cc1cnc2n1CC(C(N1CCCC1CN(C(=O)CC1(C)OCCO1)C)=O)CC2 C1(NC(CCOC)=O)CCN(C(=O)C(n2cc(C3OCCO3)nn2)C)C1 N1(C(C(c2ccnn2C)C)=O)CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)CC(F)C1 c1(C(C)NC(CCCC)=O)ccc2c(c1)CN(C(C1CC1(C)COC)=O)C2 c1(C(N(C(C)C)Cc2ccco2)=O)c[nH]nc1CNC(=O)C(C)N1CCCC1 N1(C(CCO)=O)CCC(CC(=O)OC)C1(C)C.C(C(C)C)OC c1(C(=O)NC23C(CN(C(CNC(N)=O)=O)C2)C3)scc2c1OCCO2 c1(C(C(=O)NCC2CCC(=O)N2)N(C(CC)(C)C)C)ccc(OC(C)(C)C)cc1 c1(C(C2(N(C)OC(c3ccc(C(C)(C)C)o3)=O)C(C)C2)C2CC2)cccnc1 C1(CNC(=O)C(C2CCOCC2)O)CC2CCC(C1)N2C(=O)C1=CS(=O)CCC1 C12(CNC(=O)CN3CC=CC3)CCCC1N(C(=O)CN1CC=CC1)CCC2 N1(C(C=CCC)=O)CCC(NC(c2ncsc2Br)=O)C(F)C1 Cc1cnc(C(N2CC(F)(C(=O)N(C3CN4CCC3CC4)C)C2)=O)c[n+]1[O-] c1(OCCOC)ccc(C(=O)NC(C)C(C)NC(=O)C(F)=CCCF)cc1N CCC(C)(O)C(=O)NC1CCC(CNC(C2(c3cncnc3)CCCC2)=O)C1 Cc1cccc(CC(=O)NCC(CC(C)C)NC(=O)CSC(=N)N)c1 Cc1cnc2n1CC(C(=O)NCC(O)CNC(C1(S(N)(=O)=O)CC1)=O)CC2 CCCCC(C(=O)NCC(C(=O)N(C)C(c1ccco1)C)C(C)C)N(C)C c1(C(=O)NCC2CCC(CNC(C3(C)ON=C(C)C3)=O)CC2)cccc(Cl)c1C C1(CC(N2C(C(C)NC(C3(CF)CCC3)=O)CCC2)=O)CC(C)(C)OC1=O c1(C(=O)NC(c2nncs2)C)ccc2c(n1)CN(C(C1(C)COC1)=O)CC2 C=CCCCC(C)(C)CNC(=O)C(CCC)NC(=O)C(F)C(F)(F)F C1(O)(C(=O)NC2(C)CC(NC(=O)C(c3cccc(F)c3)O)C2)CCOCC1 C12(C(N3CC4(CN(C(c5c(N)cncc5)=O)C4)C3)=O)CC1COC21CCC1 c1(C(N2CC3C(CN(C(C(CSC)(C)C)=O)C)C3C2)=O)ccc(F)c2c1CCC2 C(C(CC(F)(F)F)NC(=O)Cc1cnc[nH]1)NC(c1c(C)sc(C(F)(F)F)n1)=O n1(CC)cc(OC(=O)COCC2CC2)cn1.C12(CCSC1)C(=O)N2.C1CC1 C1(NS(CC(=O)OCC)(=O)=O)CC2CC1CN2C(C1(COCC)CC1)=O.C(C)(C)N N1(C(C(C)CN2CCOCC2)=O)CCC(O)(CCNC(=O)CCc2ccon2)C1 c1(OCC(=O)NCC(CC)NC(C2CC2(C)C)=O)c(F)cccc1F c1(CC(CC)NC(=O)C(=O)N(C2CCC2C)C)ccccc1 c1(N(C(=O)C(F)Cc2ccc(Br)nc2)C)csc2c(F)cccc12 Cc1ccccc1OC(=O)C1CC1.C(CC#N)(C(=O)N)NC(=O)OC(C)(C)C C12(NC(c3n(C)cc(Cl)c3)=O)CCCC1CN(C(C1CCCC1(F)F)=O)C2 CC1(C)CCCC(C(=O)NCC2CCCN2C(c2cnc(O)cc2O)=O)O1 C1(CC(=O)NC(c2occ(C(N(CCCSC)C)=O)n2)C)CC(=O)NC1=O C1(NC(C(CC)=CCCC)=O)CCOCC1C(=O)NOCC1CCC1 c1(C(=O)Nc2cncc(C(=O)NC(c3ccc(Br)cc3)C)c2)cc(Cl)c(Cl)nc1Cl [N-]=[N+]=NC1CN(C(c2cnc3c[nH]nc3c2)=O)CC1NC(C1(F)CCCCC1)=O N1(C(CCS(=O)(=O)NC)=O)CC(C)CN(C(=O)C(C)N(C)C)CC1C Cc1cccc2c1OC(C(=O)NCC1CCCN(C3CCCCC3)C1)C2 CCCCCC(O)CC(=O)NC1CCN(C(=O)C(O)C(C)CC)CC1C(N)=O N(C(=NCc1ccnn1C(F)(F)F)NCC(C)(C)C(C)(F)F)C(C)C CCCCC(O)C(C)C(=O)NCC(Cc1ccccc1)NC(=O)C(C)(C)CC C(C1CN(C(=O)CCSCC(C)(C)C)CC1C(=O)NCC(O)CO)=CC c1(-n2cc(C(=O)NCC3(OC)CCCCC3)nn2)ccc2c(c1)OCCO2 C1(N(C)C(c2ccncc2)=O)CCN(C(c2cc(C#N)ccc2O)=O)CC12CC2 C(=O)(CC(C(F)(F)F)NC(C1CC1Cl)=O)N(C)CC1CCC(=O)N1 C(C1COC(C)(C)O1)=CC(N1CCCC(C(=O)NCCC2CCN(C)C2)C1)=O N1(C(C=CC)=O)CCC2(CC1)CC(C)N(C(C1CCc3ncnn3C1)=O)C2 N1(C(c2c[nH]nc2Cl)=O)CCC(C(=O)NC2(CF)CCC2)C(CO)C1 N1(C(C2(CNC(=O)CCCn3ccnc3)CC(=C)C2)=O)CCC2(CCN(C)C2)C1 C#Cc1ccc(C(=O)N(C2CCN(C(c3cc(CC)nn3C)=O)CC2C)C)cc1 C1(NC(=O)OC)CCCC(NC(=O)Cc2c[nH]c(C(=O)NCCSC(C)C3CC3)c2)C1 c1(-c2nc(C3CCN(C(=O)OCC)C3C)on2)cccc(C)c1C N1(C(c2c(C(C)NC(c3ncc(NC)nc3)=O)noc2)=O)CCCC2(CC1)CC2 CC1CSCCN(C(C2CCN(C(=O)C3CC(=O)C3)O2)=O)C1 CC1(C)CC1(C)C(=O)NC.C(C)(CN)(C(=O)C=CC=C(Cl)Cl)C1CC1 N1(CCN(C)C(C2CCCC2)=O)CCN(C(C2OCCC2(C)C)=O)CC1 N1(C(c2c(C)nn(CCO)c2)=O)CC(C)(C)CC1CNC(C1CCCC1(C)C)=O N1(C(C2(C)CC2)=O)CCCN(CCNC(c2ncc(F)cc2F)=O)CC1 c1(OC)cc(C(c2nnnn2C(C)C)NCC2CCCNC2=O)c(F)cn1 C1(F)(C(=O)NCC(C(=O)NCCC2C(C)(C)OCC2)N(C)C)CCCCCC1 C12(NC(CCC(=O)OC)=O)CCCCC1CN(C(=O)CCc1cc(C)n(C)n1)C2 c1(OC)nc(=NCC2CCCC(NC(=O)C(C)CC3CCCC3)C2)[nH]c(C)c1F O=C(C1=CCCCO1)NC1CCCN(C(C23COCC(C2)OC3)=O)CC1 c1(C(=O)OC)cc(NC(=O)C(c2cnccc2C)OC)cc(N2CCNC2=O)c1 C(CCCCCC(=O)N(C)Cc1cnnn1C)NC(C(CCC)OCC)=O N1(C(C)C)N=C(C(=O)NC23CC2CN(C(c2cnn(C)c2C#N)=O)C3)CCC1=O N1(C(=O)CCc2ncccn2)CC2(CCN(C(C3CC(F)(CO)C3)=O)C2)C1 C=CCC(CC(C)C)C(=O)NC1C=CCN(C(C2CC(OCC)C2)=O)C1 c1(C(=O)NCC2CC2NC(c2ccnn2-c2ccccc2)=O)ncoc1C1CC1 c1(C(C)=O)ccc(C(=O)NC(CNC(C2(C)CC2(C)C)=O)C(C)C)s1 C1(NC(C(C)(C)OCC)=O)CN(C(=O)C(O)CC)CCC1(C)C CC1=CCC(C(=O)NC(C)C(CO)NC(=O)CSC(F)F)CC1 c1(CCC)ncccc1C(=O)NCCCOCCN(C(=O)C(C)N(C)CC1CC1)C CC1CCCC=C1C(=O)N1CC(F)CC1CNC(C1(CC(F)F)CCC1)=O c1(C(=O)Nc2ccnc(F)c2O)nc2ncc(Br)cc2[nH]1 C1(C(N2C(C)(C)CCC2)=O)N(C(=O)CSC2CC2C2(C)COC2)CC12CCCC2 N1(C(c2cn(CCC)nc2)=O)CC2(C1)CN(C(=O)CC(C)(C)CC)CC2C(=O)O C1(C(=O)NCCN(C(=O)CC(F)F)CCOC)CCn2cc(CC)nc2C1 CP(C)(=O)C1CCCC1C(N1CCC2CN(C(=O)CSCc3cscn3)CC12)=O C1(C(N(C)CC2(O)CN(C(=O)CC3CC(=O)C3)C2)=O)CC(c2ccccc2)=NO1 C(=O)(C(C(C)(C)C)NC(=O)Cc1ccns1)N(CCC#C)CCOC C(CNC(=O)C(C)(C)c1ncco1)(CC(F)(F)F)NC(c1cc(CC)[nH]n1)=O N1(c2snc(C(=O)OC)n2)CC(NC(=O)C(C)=C2CC2)CC2(CC2)C1 Cn1nncc1C(=O)NCCC(C)(C)NC(c1cncnc1)=O c1(C(N2CCC(CCNC(C3(C)CCC(=O)NC3)=O)C2)=O)nccc2nn[nH]c12 CCC#CC(C)(C)NC(C1CCC(NC(c2coc(C(C)C)n2)=O)C1)=O Cn1ccc2ccc(NC(=O)NC3COCCC3N3CCCC3)cc2c1=O N1(C(c2c(C)csc2)=O)CCCC(F)(CNC(C2CCCC(F)C2)=O)C1 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CCC2(C1)C(F)(F)C2(F)F c1(NC(C2N(C(CC(C)C3CC3)=O)C3C(C2)C3)=O)cccc2nccn12 CCCCCC(C)(C)CNC(=O)C(CN(C)C)NC(C1COC(=O)N1)=O c1(COC)nc(CC(=O)NCC2(O)CN(C(C3CCC(=O)O3)=O)C2)cs1 C1(C(=O)NC(C(C)(C)C)CO)CCC2(CC2)N1C(C12CCC(C1)C2)=O CC1CC(NC(C2CC2C(F)(F)F)=O)CCN1C(=O)C(C)C1CCCC1 C1(CN(C)C)CCCC1NC(c1ccc(NC(=O)CN(C)CC2CC2)s1)=O Cc1cc(C(N2CC(CN(C(=O)C(F)(F)Cc3ccccc3)C)C2)=O)cc(Cl)n1 C1(CNC(=O)CCOCC(F)(F)F)CCCN(C(=O)C(c2ccc(O)nc2)(F)F)C1 CCC1=C(C(=O)N2CCC3CC23C(=O)NCc2ccco2)CCCO1 c1(CC(=O)NCCCC2CCCN2C(=O)CCc2cc[nH]n2)ccc(F)nc1 C1(C)(CNC(CC2CC(SC)C2)=O)CCN(C(=O)CN(C)C)C1 N1(C(c2cc(CC)no2)=O)CCCC(O)(CCNC(c2[nH]c(C)nc2CC)=O)C1 C1(C(N2C(C)CCN(C(C34CCCCC3C4)=O)CC2)=O)CC12CCC(F)(F)CC2 C1(C(=O)N(C(C)CN(C)C(C2CC3COCC3C2)=O)C)(OC)CCC(C)(C)CC1 C#CCC(O)C(=O)NC(C)CNC(c1ccc(C(C)=O)cn1)=O c1(OC)ccc(C(N2CCC(C)C2CNC(=O)CCc2cnc[nH]2)=O)cc1 N1(C(c2c(C)cc(C)c(C)c2)=O)CC2(CCN(C(C3CCCC3(F)F)=O)CC2)C1 C(=O)(C1=CNC2=NCCC2=C1)NC1C(CNC(CN2CC(C)(C)C2)=O)CCC1 CCCC(C#N)C(=O)N1CCCCC1CC(=O)NC(C)(C)CC(F)(F)F C1(CC)CCN(C(=O)CCOC(C)=O)C1C(=O)NC(CC)C1CCC1 CC1NC(=O)OC12CN(C(C1(NC(C3CC=CCC3)=O)CCCC1)=O)C2 c1(CC(=O)OC2CCC(C(=O)OCC)CC2)cnc2ccccc2c1OC C1(C(N2CC(C(C)O)C2)=O)CN(C(=O)CC2CCCOC2)CC(C)(C)C1 C=CCCCC(=O)N1CC(C(N2CCC(C)(CC)C2)=O)(CC)C1 c1(C(C(=O)NCC(C)C)N(C)CC2CC(=C)C2)cn(CC)cn1 C=CC(O)C(=O)NCC(O)CCNC(=O)Cc1csc(C(F)(F)F)n1 C(=O)(C1Cc2ccccc21)NC(CC)CNC(=O)C(F)(F)c1ccsc1Cl C(=O)(C(F)(CNC(C1CC(=O)NC(=O)N1)=O)C(C)C)Nc1c(OC)cc(C)cc1 C12CCC(CC1)C(=O)N2.c1(CN(C)CC2C(C)CC2)occc1Br.OC c1(CN2CC(CC(=O)N(C)Cc3ccc(Br)cc3)OCC2)ccc2c(c1)CCN2 c1(CC(=O)NC2C(NC(CNC=O)=O)CC2)ccc(SC2CC2)cc1 n1(CCCNC(=NCCC)NC2CCC(CS(C)(=O)=O)CC2)cnc2ccccc12 C(=O)(CC(C)CC(C)(C)C)N1CCC(CNC(c2cncc(OC)n2)=O)(CO)C1 N1(C(c2ncn(C)c2)=O)CC(NC(C2(C)CC2(C)C)=O)C(C(F)F)C1 C(=O)(C(C)(CCC)CCC)N1C(C)CCN(C(CCCC)=O)CC1 N1(C(C(C(C)C)=O)=O)CCC(CC(N2CCN(CCF)CC2)=O)C1(C)C c12cccc(c1)NC(=O)C(=O)N2.C1(CC(=O)NC2CC2)COC2CC1C2 N1(C(C2C=CCCC2)=O)CC2CCC(C1)N2C(=O)Nc1cc(CCCO)on1 C1(C(=O)NC(CCCC)CC)CC2(CCN(C(C3CCCC3CCOC)=O)C2)C1 CC(C)C(C)CC(=O)NC(C)C(N1CCOCC(CO)C1)=O c1(C(=O)OC(C(C(=O)OC)NC(=O)OC(C)(C)C)C)ccc(C)c(C)c1F c1(C(N2CC3(CC(CNC(C(C)CN(C)C)=O)C3)C2)=O)c[nH]nc1S(N)(=O)=O C(=O)(N1CC(O)C(O)CO1)c1c(CNC(=O)CN2CSCC2=O)occ1 CCC1=C(C(=O)NC2CC(CNC(c3ccn4ccnc4c3)=O)C2)SCCO1 c1(C(=O)N(C2CN(C(c3n(CC)ncn3)=O)C(C)C2)CC)c(F)ccc(OC)c1N c1(C(N(C2CCN(C(CC=C)=O)C2)CC2CC2)=O)ncnc(C)c1C c1(OC)cnc(NC(C2CN(C(C3CCCN3C(C)C)=O)CC23CC3)=O)c(F)c1 N1(C(C(C)n2ccnc2)=O)CC2COCCC2(NC(=O)C=Cc2cncn2C)C1 N1(C(C(C(C)C)(C)C)=O)CCCC(C2CN(C(c3cc4n(n3)CCOC4)=O)C2)C1 N1(C(CC(C)F)=O)CCCN(C(C2(C)CCN(C(=O)C(O)C3CC3)CC2)=O)CC1 C1(C(=O)Nc2c(CN(C)CCCC(F)(F)F)ccnc2)CCCCNC1=O c1(-n2cc(CCC(N3CCCC4CC34)=O)nn2)ccc(Br)c(-n2cccc2)c1 N1(C(COCc2onc(C)n2)=O)CCCN(C(c2nccn2C)=O)CC1 c1(C(N2CCC(C(C)NC(CN(CCC)C)=O)C2)=O)cc(OC)cc2c1CCC2 c1(C(=O)NC23CCC(C2)N(C(C2CC4(CC4)CO2)=O)C3)ccc2[nH]ccc2n1 N#Cc1sc(-c2ccccc2)cc1NC(=O)CCCNC(=O)CN N1(C(C(C)N(S(C)(=O)=O)CCO)=O)CC(n2cc(CN(C)C)nn2)C(C)C1 N1(C(CCC(=O)NCCC)=O)CCCCC2(CCN(C(=O)C=CS(=O)(=O)CC)C2)C1 O=C(C1=CCS(=O)(=O)C1)NC1CCCC1NC(=O)C(F)C(F)(F)F N1(C(C(C)OC)=O)CC2(CCCCC2)CC1C(N1CCN(C(C)C(=O)O)CC1)=O CC1CN(C(=O)C(C)(C)N2CCCC2)CCC1CNC(=O)CCn1ccnc1 N1(C(C2C(c3cn(CC)nc3)OCC2)=O)CCC2C(CCCN2C)C1.C1CS1 Cn1cnc(C=CC(=O)NCC2(F)CN(C(=O)C=CC3CCCO3)C2)c1 CC(CNC(=O)CN(C1CC(C#N)C1)C(=O)C=Cc1ccco1)C(F)(F)F C1(NC(=O)CC2(O)CCOC2)CC2CCC1(NC(c1ccc(CF)cc1)=O)C2 C1(C(=O)NCC2CC(NC(C3(CF)CC3)=O)C(O)C2)CC2CCCCCN12 c1(C(N2CC(C#N)C3(C2)CCC3)=O)cc(Cl)cc2ccccc12 CC(C)CC(CC(=O)NC1CCC=CCCC1)NC(=O)C(O)CC(C)C C(C(C(C)C(C)C)NC(c1ccc(F)c(O)c1)=O)NC(c1cnc(OC)nc1)=O C1(NC(C(C)OCC(C)C)=O)CC(O)(CNC(c2ccon2)=O)C1 Cc1ccc(CNC(=O)CSCCNC(C2(C)CCOC2C)=O)cc1F c1(NC(CCN(C(=O)C(C(C)CC)N(C)C)CC)=O)ccc2nc[nH]c2c1 C(CC(C)C(=O)NCC(C)NC(c1cnn(-c2ccccn2)c1N)=O)OC c1(NC(C(C)(c2ccccc2)N(C)C)=O)cc(C)cc2ccoc12 CN1CC(NC(C2(NC(=O)CSc3nc[nH]n3)CC(CO)C2)=O)C(C)(C)C1 c1(C(N2CCN(C(CC(C)OC)=O)C(CC(F)F)C2)=O)coc2ccccc12 c1(CC)cc(C(=O)NCC2CC(C)N(C(c3cc(CC)no3)=O)C2)ncn1 Cc1ccc(C(=O)NCC2CC2NC(=O)CNC(=O)Cc2ccccc2)o1 c1(C(=O)NCCCC(C)NC(=O)CCN2CCOC2=O)ccc(N2CCC2)nc1 C(=O)(C(F)(F)c1cccnc1)NCC1CN(C(C(=O)NCC(F)F)=O)C1 Cc1c[nH]cc(C(=O)NCC2CCC2NC(=O)Cc2c(F)cccc2F)c1=O c1(C(=O)NC(C2CCCC2)CNC(=O)C=Cc2cc[nH]n2)nnc(O)c(Br)c1O N1(C(C2C(OCC)C2)=O)CCN(C(C2(C)CCOCC2)=O)CC1c1nccn1C c1(C(N2CC(CC)CC(O)C2)C(=O)NCCCC)cc(OC)c2c(c1)OCO2 c1(C(N2CCN(C(C3ON=C(C)C3)=O)C(CCO)C2)=O)cn2cc(C)ccc2n1 N1(C(c2[nH]cc(C)c2)=O)CCCC(CC(=O)NC(c2nncs2)C)C1 C1(NC(c2c(CC)ncnc2)=O)CC=C(C(=O)N2CC(CO)CC(C)C2)C1 Cc1c(NCc2ccnc(C(N)=O)c2)ncnc1NC1CNC(=O)C1 C1(C(=O)Nc2c(C)nsc2)CC2(CCN1C(C1OCCOC1C)=O)CC2 C(=O)(CC(C)CC(F)(F)F)NC1C(N(C(C=CC=CC)=O)C)CCCC1 C#CC1(C(=O)NC2CCCCC2C(N2CCC(OC3CC3)CC2)=O)CC(=O)C1 N1(C(c2ccc(CC)[nH]2)=O)CCC(NC(C2CCCCC2(C)C)=O)C(O)C1 C(=O)(C(CCSC)NC(C1CC(CC2CC2)C1)=O)NCC1C(CC)COC1 C1(C(=O)NCc2scc(C(N3CCC(N(C)CC)C3)=O)n2)CC2C(C1)C2(F)F N1(C(c2ccn(CC(F)F)n2)=O)CC2(CCN2C(=O)CCc2ccc(O)nc2)C1 N1(C(=O)OC(C)(C)C)CC(C)(C)C1C1CCN(C(C2(CO)CCCCC2)=O)CC1 Cc1nn(C)c2c(N(CC(F)(F)Br)C)nc(=NC3CCCc4ccc(C)cc43)[nH]c12 Cc1nccc(C(=O)NCC2(F)CCC(CNC(=O)COc3cn[nH]c3)CC2)c1N c1(C(=O)Nc2cnc(C3CCC3)o2)c[nH]c2c(F)cc(Br)cc2c1=O c1(C(=O)NCC(C(C)C)NC(C23CCC(CC2)OC3)=O)ccnc(S(N)(=O)=O)c1 N1(C(C2(COC)CCOC2)=O)CCC(C)(CC(=O)NC23CCC(C2)OC3)C1 N1(C(c2cc(C)on2)=O)CCC2CCN(C(=O)Cc3sc(C)nc3C)CC12 C1(CNC(CSCCC)=O)CC2CC(C1)N(C(c1n[nH]cc1Cl)=O)C2 C1(C)(CC)C=C(C(=O)N2CC(NC(=O)CC3NC(=O)NC3=O)C2)C1 CC1=NS(=O)(=O)NC(C)=C1CCC(=O)N(CCCN(C)C(C1(C(C)C)CC1)=O)C c1(OCC)ccc(NC(C2CCC3CC2C3)=O)cc1Cl.C1(CC(=O)N)CNCCOC1 c1(C(C2CC(OCCOC)C2)C2(O)CC2)cccc(Cl)c1 C1(O)(CCNC(c2n(C(C)C)ccc2)=O)CCN(C(C2NC(=O)OC2C)=O)CC1 N1(CCC(=O)NCCC2CC(NC(CCc3ccn(C)n3)=O)C2)C(=O)CCC1=O CC1(C)OCCN(c2nccc(C(F)(F)F)n2)C1CNC(=O)C(O)C1CC1 C(=O)(CC(C)P(C)(C)=O)N1CCC(CN(C(=O)CNC(C)=O)CC)CC1 CC(C)(CNC(=O)CC1CCCC(NC(C2CCC(O)C2)=O)C1)C(N)=O c1(C(N2CC(C(C)NC(C(CCOC)C)=O)OCC2)=O)c2ccccc2nn1C C1(CC(=O)NCC(N2CCSCC2)C)(CC)CCOCC1 N1(CC)CCN(CC(C(C)C)c2ccccc2)CC1.C12CC(C1)NC(=O)N2 c1(C(=O)NC(C2(O)CN(C(=O)CCc3cnc(C4CC4)o3)C2)C)cn(C)c(O)n1 N1(CCC)CCC(N=c2nc(N(CC(C)C)C)c3c([nH]2)c(C)nn3C)CC1 C(=O)(C1=CC(O)CCC1)N(CC(C)(C)NC(C1(NC(N)=O)CC1)=O)C c1(NC(c2ccc(C3(C)NC(=O)NC3=O)cc2)=O)ccc2c(c1)CCCC(O)C2 N1(C(c2ccc(C#C)cc2)=O)CC2C=CC1C(C(=O)N(C)CCOC)C2 C#CCCN=C(N)NCCc1cc(Cl)ccc1Br.n1(CC)cnc(-c2ccccc2)n1 Cc1ccc(N2CC(C(=O)N(CC(O)CNC(=O)CN(C)C)C)CC2=O)cc1 N1(C(=O)Cn2cc(CSCCOC3CCCO3)nn2)CCCCC1CC1CC1 CC(C)CCC(F)C(=O)N1CC2CCCC2(NC(=O)CSC2CCCCO2)C1 C=CC(C(F)(F)F)NC(=O)C(CC=CC)NC(c1[nH]cc(C)c1C)=O C1(C(=O)NCC2(NC(C3CN(S(CC)(=O)=O)C3)=O)CCCC2)OC2CCC1CC2 c1(C(C)C)nc(N2CCCC(C(N)=O)CC2)cc(N2CCC(C3CC3)C2)n1 CC(C)C(CCNC(=O)CCCc1nc(C2CC2)no1)NC(=O)C(C)N(C)C C1(C(=O)NC(CCC)c2ccco2)CN(C(=O)C(O)CCN(C)C)C(C)(C)C1 c1(C(=O)NC(CNC(c2cnc(OC)s2)=O)C)[nH]c(-c2cccc(Cl)c2)nc1C CC(C(=O)NC1CN(C(=O)CSC2CC(=C3CC3)C2)C1)(C(F)F)c1ccccc1 c1(C(=O)NC2C(NC(c3c(OCC=C)cccc3)=O)C2)cc2c(s1)CCC2 c1(-c2scc(CC(=O)NC3(CCNC(C4CCOC4)=O)CC3)n2)ccccc1F N1(C(C=C(C)C)=O)CCC2CC12C(N1CCCC1CCO)=O c1(C(C)=O)ccccc1NC(=O)C(=O)Nc1cccc(Br)c1.C12CC(C1)N2 Cn1[nH]c(C(=O)NC(C)(C)CCCNC(C2(C)CC3CC3C2)=O)nc1=O C(=O)(CC(O)CCSC)N(CC(C)NC(c1nc(OC)ccc1Cl)=O)CC N1(CC(=O)NCCN(C(C2CN3CCC2CC3)=O)CC)C(=O)CC(C)(C)C1=O C#Cc1ccc(C(=O)NCCN(C(=O)C=Cc2cc[nH]n2)C(C)C)c(C)c1 C(=O)(CC(C)(C)N(C)C)N(C1CCN(C(=O)CCc2ccccc2)C1)C N1(C(c2nn(CC)c(=O)cc2)=O)CC2CCN(C(C3CC(C)(F)C3)=O)C2C1 c1(COC)n[nH]c(=NCC(CC(C)C)NC(c2cn3cccnc3n2)=O)s1 Cc1c(NC(c2cnn(C(C)C)c2Cl)=O)cccc1N1C(=O)CCNC1=O C1(NC(CN(C)S(N)(=O)=O)=O)CN(C(c2cnn(CCO)c2)=O)C2(CCOC2)C1 N1(C(C(C)CN(C)C)=O)CCC(OCCNC(C2CC23CCC3)=O)CC1 N1(C(C(C)NC(N)=O)=O)CC2(C1)SCCC2NC(=O)CC1=CCOCC1 CN1CCN(C(c2cnsn2)=O)C(C(N2CCC(O)C2)=O)C1 N1(C(c2nc(C(N)=O)sc2)=O)CCC2(CC1)CC2CNC(=O)C=CC1CC1 N1(C(CC(COC)C)=O)C2CCC1C1CC1(NC(c1cnc(C)s1)=O)C2 c1(C(=O)NCC(C2CCC2)NC(C(n2ncc(C)c2)C)=O)ccc(Cl)cc1F C(=O)(C(F)(F)CCn1ccnn1)NC12CC(CNC(C(C(C)C)SC)=O)(C1)C2 c1(OC)cccc(C(=O)N(C)CCN(C(=O)Cc2ccccc2SC)C)c1OC C1(C(=O)NCCN(CCCC)C)C(C2CC2)CCN1C(c1ccc(O)cc1F)=O C1(COCC)CCCN(c2cc(N3CCC(C)=C(C)C3)nc(CC)n2)CC1 N1(C(C2(OC)CCN(C(c3nc[nH]n3)=O)C2)=O)CCC(C)C(F)(F)C1 N1(C(C2CC(=O)C2)=O)CC(F)(CNC(=O)CCn2cncn2)C1 c1(C(N2CCN(C(CC(CC)C(C)C)=O)CC2CO)=O)cc2cc(C)ccc2[nH]1 c1(CC)nc(C)oc1C(N1CCOCC1c1noc(C(=O)O)n1)=O c1(C2C(C(=O)NCC3(CNC(C(C)SC)=O)CCC3)C2)ccnn1C N1(C(C2CC(C(=O)OC)C2)=O)CCCC2CN(c3ccc(S(C)(=O)=O)cn3)CCC12 Cc1ccnc(C(N2CCCC(CO)(CNC(C3(CCC(C)C)CC3)=O)C2)=O)c1N N(C1CN(C(c2c(C)[nH][nH]c2=N)=O)CCc2ccccc21)C(C(CSC)(C)C)=O c1(CN2CC3C(C(=O)Nc4c(OCC)cccc4)(C3)C2)ccc([N+](=O)[O-])c(F)c1 C1(C(=O)NC(C)CC(=O)NCCC2(C)CC2(F)F)COCC1(C)C N1(C(C2CC(Cc3ccccn3)C2)=O)CCOCC1CC(c1cccc(O)c1)O N1(C(C2(F)CCN(C(C3(C)CC=CC3)=O)C2)=O)CCCC2(CC1)CC2 c1(NC(c2nc(C)[nH]c2Br)c2n(CCCC)nnn2)ccc2c(c1)CN(C)C2=O C(CCCC(C)(C)NC(C12CCC(C1)C2(C)C)=O)NC(c1ccnc(C)n1)=O CC1CC2(CC(C(=O)NCC#CC(=O)Nc3ccc(=N)[nH]c3)C2)C1 C=CC1(C(=O)Nc2ccn3nccc3c2)CCN(C(=O)Cc2cc(C)cs2)CC1 N1(c2snc(COC)n2)CC2(CCCC2NC(c2coc(C(C)C)n2)=O)C1 N1(CCN)CCC2(CC1)CC2C(F)(F)F.N1(C(=O)OC(C)(C)C)CC(C(=O)O)CC1CO c1(NCc2ccc(CNC(C3C(C)N(C)CC3)=O)cc2)ccc(Cl)cc1C(N)=O C(=O)(CC1COc2ccccc21)NC(C1(O)CN(C(CC=C(C)C)=O)C1)C c1(CC(=O)NC(C(=O)OC)CO)ccccc1OC(F)(F)F c1(C(N2CCC(NC(CCCCC)=O)C2)=O)ccc(C)c(C(C)=O)c1 C1(CONC(=O)CC2CCCCN2C(=O)Cc2cc[nH]n2)CC2C=CC1C2 c1(SC)nc(C(=O)NCC#CCNC(=O)Cc2cc(C)on2)cs1 c1(NC(c2nnc(O)o2)C)cc(N(C)CC2(c3cccs3)CCCCC2)ncn1 C(=O)(CCN(OC)C(=O)C1(N(C(=O)C(OC)OC)C)CC1)OC C(C(C)(C(C)C)NC(=O)C(C)CN1CCCCC1)NC(CC1CC(SC)C1)=O c1(C(N2CCC(CC(C)C)C2)C(=O)NCCC)cc2n(n1)CCCCO2 Cn1ccc(CC(=O)NCCC2CCC(NC(c3csc(S)n3)=O)C2)n1 C1(Cc2ccccc2)(SCCCOC2CC2)CCNCC1 C1(C)(NC(COCCC=C)=O)CCN(C(=O)CC2CCC(CC)O2)CC1.C(C)(C)C N1(C(Cc2[nH]c(=NCC)sc2)=O)CCC2(NC(=O)C=CC=C(Cl)Cl)CCCC12 Cc1ccc(C(=O)NC2CCCC2NC(c2ncccc2C(F)(F)F)=O)c(F)c1 N(C(=NCCOc1cccc(Cl)c1)NC1CCOC1C)C(CC)CC c1(C(=O)NC(C)Cn2cc(CCN(C)CCO)nn2)ccc2c(c1)NCCC(=O)N2 c1(C=O)ccc(OCF)cc1.C1(CCC(=O)N(C(C)=O)CCO)CCC(C)O1 c1(CC)cccc(NC(=O)CC(CNC(c2cnn(C(F)F)c2)=O)OC)c1 c1(C(N2CC(C(C(=O)N(CCCC)CC(C)C)O)C2)=O)cc[nH]c(=N)n1 Cc1ccnnc1C(=O)NC1CC(CNC(=O)C(F)(F)c2csc(Cl)c2)C1 Cc1cc(=NCC(C)c2ccncc2)[nH]c(=NCCN2CC3CCC2C3)[nH]1 C1(NC(c2cncc(C)n2)=O)CCN(C(C2CCCN2C(=O)N(C)C)=O)C12CCC2 N1(C(C(=O)Nc2cn(CC)nc2C(C)C)=O)CCCC2NCCCCC12 Cc1ccc(C(=O)NC(CC(=O)NCC(c2ccccn2)O)C2CC2)cn1 C12(NC(C=CC(CC)C)=O)CCCC1N(C(=O)Cc1nnc(S)n1C)CCC2 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CN(C(=O)CC1C=CCC1)CCO2 C#CCC(C)(C(=O)NC(CO)CC#CC)NC(=O)COC1(C)CCC1 c1(C(=O)NC(CNC(C2(OC)CCCC2)=O)CO)cc(C)c(-c2cccs2)s1 C1(NC(c2cc(C(F)(F)F)no2)=O)CCSC12CN(C(C1CCS1(=O)=O)=O)C2 c1(-c2ccc(C(C(=O)NC3CCC3)N(C(C)C3CC3)CC)s2)cccc(Br)c1 Cn1cc(C(=O)OCC2CCC(N(C)C)CC2)cc1C(F)(F)F Cc1cccc(C)c1C1(O)CCN(C(=O)C=Cc2ccc(Cl)cc2)C1 CC(C)C(CNC(c1cccc(C(=O)NCc2cn(C3CC3)cn2)n1)=O)C(C)C N1(C(C2(CC(=O)OC)CC2)=O)CCCC(NC(c2ccc(C)c(O)c2)=O)C1C CCC(CC1CCCCC1)C(=O)NCC(C)CC.c1(C(=O)N)ccccc1CSC Cc1cnc(F)c(C(=O)NC2CC(C)N(C(C3CN(C4CCCCC4)C3)=O)C2)c1 CN1CCCC(C)(C(=O)N(C2(CC(=O)N3CCC3)CC2)C)C1 N1(C(c2cncc(CNC(CC3CCC(C)C3)=O)c2)=O)CC2CCC(C1)C2O C1(CC(=O)NC(C2CCCCC2)CNC(=O)C=C2CCCCC2)CCC12CCC2 c1(C(N(C(C)CCNC(c2cnnn2C2CC2)=O)C)=O)ccn2nccc2c1 c1(CCC)ccc(C(=O)N(CCNC(=O)C(C)(COC)OC)CC)cc1 C(=O)(CCS(C)=O)NCCCC1N(C(COCCOC)=O)CCC1 c1(C(=O)NC(CC)CNC(C2CCSC2)=O)cccnc1C(F)F C1(CNC(C2(C)CCOCC2)=O)CC2CCC(C1)N2S(=O)(=O)CCC(F)(F)F c1(C(N2CCN(C(C(CC=C)C)=O)CC2CF)=O)ccc(F)c(S(C)(=O)=O)c1 C1(CCC(=O)NC(CNC(C2(CC=C)CC=CC2)=O)CC)NC(=O)NC1=O N1(C(CSCC)=O)CCN(C(=O)Cc2nc(C(C)(C)C)cs2)C(CC(F)(F)F)C1 C#Cc1ccc(C(=O)NC2(CO)CN(C(=O)Cn3cc(C4CC4)cn3)C2)c(F)c1 c1(CC(N2CC3N(C(C(CC)OCC)=O)C(CC3)C2)=O)ccc2ccccc2c1 C=CCCC(C(=O)NCc1cc(C)n(CC)n1)NC(=O)CC1CC(C2CC2)C1 Cc1cc(C(N2CCN(C(c3cccc(Cl)c3Br)=O)CC23CC3)=O)c(F)cc1Br Cc1ccc(C(F)F)c(C(N2CCC(C)(NC(c3cnc(C)cn3)=O)C2)=O)c1 C12(CNC(Cn3c(C)cc(C)n3)=O)CN(C(=O)CN=S(C)(C)=O)CC(F)(C1)C2 C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(=O)C(C)SC)CC(OC)C1 CC1(CNC(=O)Cc2cnns2)CCCN1C(c1cccn1C1CCCC1)=O C1(NC(c2ccc(OC)c(OC)c2)=O)CC2CC(C1)N(C(C1CC3(CC3)C1)=O)C2 CS(=O)(=O)CCCC(=O)NCC1CN(C(=O)Cc2ccccc2Cl)CC12CC2 C1(C(=O)NC(COCC#C)C)(CC)CCN(C(=O)CCOC2CCC2)C1 N1(C(c2n(CC)ncc2)=O)CCC2(CC1)CC2C(=O)NC(c1ncccn1)CC C1(CCC(=O)N2CCC(c3cnco3)C2)CC(=O)CN1C.C=CCC(=O)OC C1(C#N)(C(=O)NC(C(=O)NC(c2n(CC)ccn2)C)CN(C)C)CC(C)C1 c1(C(=O)NCCNC(C2(CCC)CC2)=O)coc2c(Br)cccc12 c1(C(C(=O)NCC(C)CNC(c2ccc(F)o2)=O)(F)F)cccc(Br)n1 c1(C(=O)NCC(C2CC2)NC(=O)CC2(O)CCCOC2)ncnc2ccsc12 CC(C)C(O)C(F)(F)C(=O)Nc1cccc(=O)o1.C123CC(C1)(C2)CNC3=O N#Cc1c[nH]cnc1=NC1CCC(NC(C2CCCC2)=O)CC1 c1(-c2cc(-c3onc(CS(=O)(=O)CC4CC4C4CCCC4)n3)n[nH]2)cccc(F)c1 C(C(C(=O)NCCN1CCCOCC1)C(C)(C)C)NC(c1c(C)scc1)=O C(=O)(C(C)CCCC(C)=O)N(C1C(=O)NCC1(C)C)C(CCCC=C)=O C1(CC)C(CC(=O)NCC2(NC(=O)C(c3ccccc3)F)CCCC2)C1(F)F O=C1CCC(C(=O)NC2C=CC(C(=O)Nc3ccccc3C(F)(F)F)C2)=NN1 c1(CN(C)CC2CCN(C(=O)C=CC3CCCO3)C2)nc(C(C)(C)C)no1 c1(CC)cc(Br)ccc1C(N1CC(NC(c2ccc(OC)cn2)=O)C(O)C1)=O c1(SC)cn(C)nc1C(=O)NCC(C(C)(C)C)NC(=O)CCCCOC(C)C Cn1cc(Cl)cc1C(=O)NCCC(=O)NC(=O)NC(c1c(CC2CC2)cco1)=O CCC(C)C(CC(=O)NCc1coc(C)n1)NC(=O)CC1CSCCO1 N1(C(c2ccc(C(=O)OC)o2)=O)CCCCC1C1CCCN(C(=O)C(C)OC)C1 C(=O)(CCC1=NNC(=O)CC1)NCC12C(CN(C(C(=O)NC(C)C)=O)C1)CC2 N1(C(c2cc(C)[nH]n2)C(=O)NCC2CCCO2)CCC(O)(c2cc[nH]n2)C1 c1(C(=O)NCC2CCCCN(C(C3CC(OC)C3)=O)C2)cn2ccccc2n1 C1(NC(CCCOCCOC)=O)CCC(CC(C)NC(=O)C=CC(C)C)CC1 c1(OC)cc(CSc2ccc(F)nc2)ccc1OCCN(C)C N1(C(CCc2c(C)n(C)nc2)=O)CCCCC(NC(=O)C(C)(C)CO)C1 C1(C(N2CCN(C(C=NOC)=O)C(C(F)F)C2)=O)CCOC2(CCC2)C1 C(=O)(C(C)S(N)(=O)=O)NC(CC)CN(C)C(C1CCS(=O)CC1)=O c1(OC)cc(C(N2CC(NC(=O)C(C)CC3CC3)C(C)C2)=O)cc([N+](=O)[O-])c1 c1(C(=O)NCC2N(C(C3C(COC)(COC)C3)=O)CC2)cc(C)c(F)cc1F C1(CC=C)(NC(C2CC(CC)=NO2)=O)CCCN(C(=O)C(CC)CO)C1 CCCN=C(NCC(O)COCC)NC1CCCC(c2ccccc2)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCC(C)NC(c1nc2ccccc2[nH]1)=O C12(NC(C3(C=C)CC3)=O)CCN(C(=O)CCCc3csc(=N)[nH]3)CCC1C2 CC1=C(CNC(C2CC23CCN(C(c2n[nH]cc2Cl)=O)C3)=O)COCC1 N1(C(C=C(COC)C)=O)CCC(C(=O)Nc2ccsc2)CC(C)(C)C1 C(=O)(C(CC1CCCCC1)CC)NC(c1cn(CC2C(C)C2(F)F)nn1)CCC c1(C(N2CC(CC)N(C(=O)Cn3nnc(C)n3)CC2)=O)nccc2ccn(C)c12 C(=O)(C1CC=Cc2ccccc21)NC1CC(CNC(c2csc3cncn23)=O)C1 c1(OC)c(C(=O)NCCC2CN(C(c3ccon3)=O)CC2C)ccnc1Cl c1(OC)cnc(CNC(=O)CCC2CCCN(C(c3cc(OC)cs3)=O)C2)cn1 N1(CC(=O)N(c2cccc(OC(F)F)c2F)CC)CCc2cc(C)cc(C)c2C1 C12(CNC(C3(C=C)CCC3)=O)CCC(CN(C(=O)CCC(CC)CC)C1)C2 c1(C(=O)NC2CC(C)N(C(C3(C4CCC4)CC3)=O)C2)c([N+](=O)[O-])cnn1C CC1(C)C2CCC1(C(=O)NC1(C)CCN(C(C3COC4COCC34)=O)CC1)CC2 c1(C(N(CCNC(C2C(CC)C2)=O)CCOCCO)=O)ccc(Br)c(C)c1 c1(OCCn2cc(C3(S(N)(=O)=O)CC(CBr)C3)nn2)cc(F)cc2c1OCOC2 CC1(C)CN(C(C2(C#N)CCC2)=O)CC(CNC(c2cncc3nc[nH]c23)=O)O1 C1(NC(c2cncc(Cl)c2)=O)CCCCN(C(C2(CCF)CCOCC2)=O)C1 OC1CCCCCC1c1cn(-c2cc(Br)cs2)nn1 CCCC(C)CC(=O)NC(C)Cn1cc(-c2cccc(F)c2)nn1 N1(C(CNC2CCCC2)=O)CC2CC1CC2NC(c1cc(C(C)C)ncc1)=O C(=O)(C(C)CC(=O)NC1(C)CC(C(N2CCOC(C)(C3CC3)C2)=O)C1)OC Cn1cc(NCc2ccc(I)cc2)cc1C(=O)NCc1ccc(F)cc1 C1(F)(CCNC(Cc2c(OC)nccc2)=O)CCN(C(=O)C(=O)NC2CC2)CC1 C(=O)(C1=C(C)CCCC1)N1CCC(CNC(C2(C(F)F)CC(=C)C2)=O)C(C)C1 C(C1=COCCC1)(c1n(CCCCCC)nnn1)NC1CCOC(CC2CC2)C1 c1(C(N2CCC(C)(C)C2CNC(=O)CC2CC3CC3C2)=O)ccc(F)c(C#N)c1 C(C(C)(C)C(C)(C)C)NC(CN(C(=O)CN1CCCC1CO)CCOC)=O N1(c2nc(C)nc(C#N)c2)Cc2nccn2CC(NC(c2ccc(Cl)o2)=O)C1 C(=O)(C(F)(F)C(F)F)NC1(C)CCN1C(=O)CN.N12CCCC1CC2=O C(C(C)CCCO)NC(C1(CNC(c2cc(Cl)n[nH]2)=O)CC(=C)C1)=O O=C(CC(C1CC1)NC(c1ccc(CO)o1)=O)NC1CCCSC1 C12(NC(C3CC3c3ccc(F)nc3)=O)CCCC1(F)CN(C(C1C=CCC1)=O)C2 c1(NC(C2C=CCN(C(=O)C=CCO)C2)=O)cnc2[nH]cnc2c1 C=CC(C)(CCOC)C(=O)NC(CC)CCCC(=O)NCc1ncnn1C(C)C c1(OC)ccc2c(c1)C(N(C)C(c1csc(CO)c1)C(=O)NCC1CC1)CCC2 C1(C(=O)OC)C(F)(F)C12CC(COC(c1cccc(CCN3CCCC3)c1)=O)C2 C1(NC(CCN(C(C2(C#C)CC2)=O)C(C)C)=O)CC(=O)N(O)C1 c1(C(=O)NC2CCN(C(C(C)OCC)=O)CC2)ccc(Br)c2c1OCCC2 C1(NC(C2OCCN(C(CC(C)=C(C)C)=O)C2)=O)CCCCCC1(C)C Nc1c(F)c(C(=O)NC2CC2NC(c2cnn3c2OCCC3)=O)c(F)c(F)c1F C1(NC(CCCC(N)=O)=O)CC2CCCC(C1)N2C(=O)CC1(O)CCCOC1 c1(C(=O)NCC(CNC(=O)C(C)C2CCC2)OC)ccc(-n2cncn2)nc1 C12(C(N(CCN(C(c3c[nH]ccc3=O)=O)CC)CC)=O)C3CCC(CC13)C2(F)F c1(C(=O)NC2CN(C(C3(CC=C)CCOC3)=O)CC2CC)ccc2sncc2c1 Nc1cc(Br)ccc1CNCc1ccc(F)cc1 c1(OC)cc(C)c(-c2cn(CCN(C(=O)CN(S(C)(=O)=O)C)C)nn2)cn1 CCCC(CCC)C(=O)N1CCC(CNC(c2ccc(Br)c(C)c2F)=O)C(F)(F)C1 C12(C(=O)NC3CCC(CNC(=O)CC4COCCO4)C3)CCCN(CC1)C2 O=C(CCCCn1ccnc1)NNC(=O)NC1CCCC1CCO CCCC(C(=O)N1CC(C2CN(C(=O)CC3CC=CC3)C2)C1)C(C)C N1(C(c2c(C)coc2C)=O)CC(NC(=O)Cn2ncc(C#N)c2N)CCC1C N1(C(c2cnc(CC)s2)=O)CC(CCOC)CC1CNC(=O)C(C)C1CCCO1 Cc1cc2[nH]c(=O)c(C(=O)NCC3(O)CCN(C(C4CC4F)=O)C3)cn2n1 c1(NC(CN(C(COC)=O)C)=O)ccc(C(=O)NC(C)C(C)(C)CO)nc1 CCC(C)(CC(=O)NC1CCC1CNC(=O)C=Cc1ncco1)C(=O)OC c1(C(=O)NC(C(C)OC)C)c(C)sc(C)c1Br C1(NC(CCC2C(C)(C)C2)=O)(CO)CCCN(C(=O)CC2CCSC2)C1 C(=O)(CC(C)C(F)F)N(C1CC2CC1N(C(c1cncc(N)c1)=O)C2)C C=CCCCCCC(=O)NCC1CC1NC(c1ccc[nH]1)=O CC(C)C(C(=O)NCCN(C1CCCC1)C(=O)C=Cc1ccc(Cl)s1)NC(N)=O C12(NC(C3CCCC(F)(F)C3)=O)CCCC1CN(C(C1CCCC1)=O)C2 N1(c2nc(C)nc(SC3CCOC3)c2)CC2CC1CN(C(=O)OC(C)(C)C)C2 Cc1oc(C(C)C)cc1C(=O)N(C1(Cc2cn(C(C)(C)C(=O)O)nn2)CC1)C N1(C(C(C2CC(F)(F)C2)OC)=O)CCCC(CCNC(=O)C(C)=C(C)C)C1 C1(NC(CCOc2ccc(CC)cc2)=O)CCC(C)N(C(c2coc(Cl)n2)=O)C1 N1(C(CCCC(CCC)C)=O)CC2CCC1C1CN(C(=O)C(O)C3CC3)CC21 C1(CC(N2CC3CC2CN3C(=O)CCCCC(F)F)=O)CCc2ccccc2C1 C(=O)(C(C)C(O)C(C)C)NCCC1CCN(C(Cc2c(OC)ccc(C)c2)=O)C1 C(=O)(C1=NNC(=O)CC1)N1CCN(C(CNC(C2(C)CCCO2)=O)C(F)F)CC1 c1(C(C)C)nnc2n1CCCC2NC(=O)NC1CC(CF)C1 C(CC(C(C)(C)C)NC(C1COCC1(C)C)=O)N(C)C(c1cc(Cl)n(C)n1)=O c1(NC(=O)C2CC2)ccc(-c2cn(CC3CCN3C(CCC)=O)nn2)cc1 c1(OC)ccc2[nH]c(C(N3CCOCC3C(=O)O)=O)cc2c1Cl CN1CCC(CC(N2CC=CC(C(=O)NC3CCCOC3)C2)=O)CC1 C1(NC(c2scc(COC)c2)=O)CCCCN(C(=O)CCn2cccnc2=O)C1 c1(C(=O)Nc2nc(NC(c3cc(OC)ncc3)=O)n(C)c2)cc(Cl)cc(Cl)c1Cl C1(NC(CN2CCC(C)C2)=O)CN(C(c2cnc(O)cc2N(C)C)=O)CC1(C)C CC(C)C(COC(=O)COCC1CCCO1)CCOC(=O)Cc1ccon1 C=CC1CN(C(CC(c2cccs2)NC(=O)OC)=O)CCO1 N1(C(CCCC#C)=O)C(C)CC2CN(C(=O)Cc3cccc(C#C)c3)CC12 C1(CNC(C(CC(C)C)N(C)C)=O)CC2COCC2N1C(=O)Cn1cnnc1 C#Cc1ccc(C(=O)NC2CC(CCNC(C3(O)CCCCC3)=O)C2)c(F)c1 c1(C(=O)NC2CC(C)(C)N(C(c3cnncc3O)=O)C2)ccn2nnnc2c1 N1(C(S(=O)(=O)NC)=O)CCC2(CC1)CCN(C(C1(C)CCNC1=O)=O)CC2 C1(C(N(C)CC2(O)CN(C(=O)C(=O)NCC3CC3)C2)=O)CCC(F)(F)CC1(C)C N1(C(CCN(C2CCOCC2)C)=O)CC(N(C(=O)CCC(C)(C)C)C)C2(CC2)C1 CC(C)CC(C(=O)NCc1ncoc1C(C)C)NC(=O)Cc1ccccc1O N1(c2ncc(CN(C)C)nc2)CCN(Cc2ccc(Cl)cc2)C(C)(C)C1 C(=O)(C1=CC2CCC1C2)NCCCC(C)(C)NC(C(C)OC)=O c1(C(=O)OCC)ccc(C(=O)NC2(CC(=O)NC3(O)CCC3)CCC2)cc1 c1(C(=O)NCCC2CCN(C(c3cc(F)c[nH]3)=O)C2)ccc([N+](=O)[O-])cc1Cl CP(C)(=O)CC(=O)NC(C(=O)NC(CCO)C(F)F)C1CC1 C1(NC(C(COC)(C)C)=O)CC2(C1)CN(C(=O)C(C)n1cccn1)C2 C(=O)(C1=CC2CCCCCC12)NCCCN(C(C(SC)SC)=O)CC1CC1 N1(C(C2CC(n3cc(CNC=O)nn3)C2)=O)CC2COCC(C2)C1 Cc1oc2ccc(CNC(=O)COCCO)cc2c1-n1cc(COC(C)C)nn1 C(C(=O)OC(C)(C)C)(C(=O)NCCC(C)CCNC(C1(C2CC2)CC1)=O)OC c1(NCCC=C=C)ccc(S(=O)(=O)NCC2CC2(Br)Br)cc1F c1(C(=O)OCc2noc(CO)n2)cc2cc(Br)ccc2nc1Cl CC(C)(C(=O)NCCCN(C(C1CCNC1=O)=O)C1CC1)C(F)(F)F c1(C(=O)NC(CNC(COCCCOC)=O)CC(C)C)oc2ccc(Cl)cc2c1C N1(C(C(CNC(C)=O)N(C)C)=O)CC2(CCCN2C(=O)C(c2csc(C)n2)=O)C1 S(=O)(=O)(c1c(F)c(F)c(F)c(F)c1F)N1CCC(C(N2CCCC3CCCCC23)=O)C1 CC1(C(=O)NCC2CC3C=CC2C3)CCN(C(c2cnc(O)o2)=O)CC1 C1(NC(C2(CCC)CCC2)=O)CC2CC1CN(C(c1ncnn1CC)=O)C2 C1(NC(c2n[nH]cc2[N+](=O)[O-])=O)CC2CC(NC(C3CCCS3(=O)=O)=O)CC12 C(C(CCC)C(=O)NCCCN1CCC(O)C1)NC(CCOCC#C)=O C(CCC(=O)N(C)CC1CCCN1C(=O)Cn1cnc(C(F)(F)F)c1)OC n1(CC)ccnc1CN(C(=O)C(C)(C)C1CCN(C(=O)C(C)NC=O)C1)C Cn1ccc(C(N2CCC(C(F)(F)F)C(NC(=O)Cc3cncs3)C2)=O)cc1=O C=CC1(C(=O)NCCC(=O)NCC=CCNC(=O)C(C)C)CCOCC1 C1(NC(c2cn(CCC=C)nn2)=O)CC2CC1CN(C(c1cscc1F)=O)C2 C(C)(CCC(=O)Nc1cccc(Cl)c1)NC(c1c(COCC)cco1)=O c1(OC)ccccc1CC(N1CC(N(C)C(C2CCSC2)=O)C1)=O N1(C(c2nc(-c3c(C)nn(C)c3)sc2)=O)CCN(C)C(c2ccc(F)s2)C1 C1(C(=O)NCc2ncc(OC)nc2)CC2(CC2)CN1C(c1ccc(C#N)cc1)=O c1(C(N2CC(C(C)NC(c3ccncc3C3CC3)=O)C2)=O)c(F)ccc(Cl)c1F N1(C(C2(SCC)CC2)=O)CC2CCCN(C(=O)Cc3cccnc3)C2C1 C12(C(N(C)CCO)=O)CCN(C(=O)C(=Cc3cccnc3)F)CC1C2.C1(=O)CCN1 C#Cc1cc(C(=O)NCC2CC2CNC(=O)Cc2ccno2)ccc1C C1(C(C)C)CC(CO)CCO1.C12CC(C)(C1)NC2=O.c1(C(=O)N)ccncc1 N12CCC(C1)CCC2=O.C(C)(C(=O)NCCOCC(C)C)NC(=O)OCC N1(C(COCCC#C)=O)CC2CCN(C(C3CC(C)(CC)C3)=O)C2C1 C(=O)(C1CCCn2nccc21)N1CCC(=CCNC(c2cnncc2O)=O)CC1 C12(CNC(c3ccc(CO)o3)=O)CCCCC1CN(C(c1csc(O)n1)=O)C2 N1(C(CC=C)=O)CCC2(CCN(C(=O)C(CC)NC(N)=O)C2)C1 O(NC(=O)C(C)OCCNC(C1CN2CCC1C2)=O)CC1CC(=C)C1 C12(CC)CC(C1)N(C(=O)C(CC1CCCC1)CNC(=O)OC(C)(C)C)C2 c1(OC(C)C(=O)NCC2CN(C(C3CCCCC3O)=O)CCO2)ccccc1Cl c1(C(=O)NCC2C(C)CN(C(=O)CCc3cncnc3)C2)ccnc2cc[nH]c12 Cc1cc(NC(c2snc(C)c2N)=O)ccc1NC(=O)CC1CC(F)(F)C1 C(CC(C(C)C)NC(c1cn(C(C)C)nn1)=O)N(C(CCN(CC)CC)=O)C C(=O)(CS(=O)(=O)C1CCCC1)NC1CN(C(CCCOCCC)=O)CC(F)C1 N1(C(c2c(SC)cnn2C)=O)CC2CCC1CN2C(=O)COc1ccccc1O Cc1csc(=O)n1CC(=O)NC1(CO)CCN(C(C2CCC(C)(C)C2)=O)C1 C12(C(N(C(c3onc(C)n3)C)C)=O)CC(CO)(CN1C(C1(F)CCOC1)=O)C2 Cc1cc(=NC(=O)CNCC(C(F)(F)F)n2cccn2)[nH]o1 C1(N(C(=O)COC(F)F)C)CCCCN(C(c2cc(C(N)=O)co2)=O)C1 C1(C(N2C3(CNC(CN(S(C)(=O)=O)C)=O)CC(C2)C3)=O)CCCCC12CCCO2 C=C1CCN(C(c2cn(CC)nn2)=O)C(C(N2CC(CO)C2(C)C)=O)C1 c1(CCCC(=O)NCC2CC(CNC(C3CCO3)=O)C2)ccc(C(F)(F)F)cc1 Cc1nn(CC(=O)NC2(C)CCN(C(=O)CSC3CCCO3)C2)c2ncccc12 n1(CC(=O)N(CCCNC(c2ccc(C)s2)=O)CC)cnc2ccccc12 N1(C(=O)NC2(C(F)(F)F)CCC(=O)NC2)CCCC(OC2CC2)CCC1 c1(C(C(=O)NC2C(NC(c3conc3C3CCC3)=O)CCC2)O)ccc(F)cc1 c1(NC(=O)NCC2(COC)CCOC2)cc(C)cc2c[nH]nc12 Cc1c2sc(c1Cl)NS2(=O)=O.Cc1nn(C(C)(C)C)c(C)c1Br.C(C)(C)(C)NC(=O)OC C=CCC(C(=O)NCC(CNC(=O)CN1OC(C)CC1=O)OC)NC(C)=O N1(C(CSc2n(C)nnn2)=O)CCN(C(C2CCC(C)(C)C2)=O)C2CCCC12 C1(N(C(C(CO)NC(C2C(C)CC=CC2)=O)=O)C)CCC(=O)N(C)C1 C(CCO)(CC(C)C)NC(C1C(OC)CN(C(c2nscc2C)=O)C1)=O C1(C(N2C(CC(=O)NCCCCCC)CCCC2)=O)OCCCC1(C)C N1(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CCN(C(C2CC2F)=O)C(CO)C1 CC1(C)COC(C(N2CCC(NC(=O)CC3CC4C=CC3CC4)C2)=O)CO1 c1(C(=O)NCC2CCCCN(C(c3ccc(CC)[nH]3)=O)C2)ncccc1[N+](=O)[O-] c1(NC(C=CCNC(C2(CSC)CCC2)=O)=O)ccn(C(F)F)n1 C123CCC(CC1NC2=O)C3.C1(C(N2C(C)(CCO)CC2)=O)CCCN1C=O N1(C(=O)Cc2cccc(F)c2F)CC(NC(C2C(C)(COC)C2)=O)C(C)(C)C1 C(N=c1[nH]c2ccc(Cl)cc2s1)C1CCC(NC(=O)C=Cc2ccccc2F)C1 Cc1ccc(OC(CNCC(=O)N(C)CC)CC(C)C)cc1.C12(CC1)C(=O)NC2.CF c1(C(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC23CC3)cccc(S(C)=O)c1 C(=O)(C(C)C(C)(C)C)N(CC(C)NC(c1cnc(CC)[nH]1)=O)C CCC(CN(C)C)CC(=O)NC1CC(C(=O)NC23CCC(C2)OC3C)C1(C)C c1(CCC(=O)NC2CC(NC(C3C(C)(C)CCO3)=O)C2)cccc(Cl)c1Cl CC(CCCCCO)NC(C1C2CC1N(C(=O)CC1(O)CCCCC1)C2)=O N1(C(C2N(C(C(n3ncc(C)c3)C)=O)CCC2C)=O)CC2(CNC(=O)N2C)C1 c1(CC2N(C(C(C)Oc3ccccn3)=O)CC=C2)ccc(Cc2nccs2)cn1 C1(CCCN(C(CCC)=O)Cc2cccnc2)CCN(C(=O)C2=CCOC2)CC1 C(=O)(CCCc1cccnc1)N(CC(CNC(C(C)SCCC)=O)O)C N1(C(c2n(CC)ncc2Br)=O)CCC2CCC(NC(=O)CC(C)(C)C)C1C2 c1(CCC)cc(C(=O)NCc2c(C3CN(C(C4CC4(C)Br)=O)C3)ocn2)sc1C C1(C(=O)NCCC(C)CCO)C2CC3C(C2NC(=O)C(c2ccnn2C)C)C13 c1(OC)ncc(SC)cc1NCC1CCCC1Oc1ccccc1 C1(CNC(c2n(CC#C)ccc2)=O)COCCN1C(=O)CCc1nc(=N)[nH][nH]1 c1(C(N2CC=CC(NC(c3cocc3Br)=O)C2)=O)cc2ccccn2c1 c1(C(=O)NC(C(CO)NC(CC(C)n2cccc2)=O)C)cc2sccc2[nH]1 CN(OC1CCCC1)C(=O)CC1(N(C)C(=O)Nc2cc(C#N)cs2)CC1 C1(NC(C2C=CCC2)=O)CN(C(c2cc3cccc(Cl)c3s2)=O)CC2(CCC2)C1 CC1=NOC(C(=O)NC(C)CCCNC(=O)CCC2CC(F)(F)C2)C1 N1(C(c2cc(COC)on2)=O)CCC(N(C(=O)C(C)C(C)C)C)CC1 c1(C(=O)NC(c2cnc[nH]2)C)ccc(-c2cncc(N)c2)cc1 N1(C(CCSCC(C)C)=O)CCN(C(C2OCCOC2C)=O)C(c2ncc[nH]2)C1 N1(CC2CCC(OC)CC2)CC2CC1CN2C(=O)OC(C)(C)C C1(CC)(NC(=O)CC(C)CNC(=O)C=Cc2cnccn2)CCCCCC1 N1(C(=O)C=CC2CCCC2)CC2(CCN2C(=O)Cc2c(F)cccc2F)C1 C1(C(=O)NC2(CC)CCCN(C(=O)COC3CC3)C2)CCc2ccnn2C1 c1(NC(C2N(C(C(C)OCC=C)=O)CC(O)C2)=O)cncc(Br)c1C c1(C(=O)NC(C2CCOC2)CNC(C2CC(OC)C2)=O)coc(Br)n1 N1(C(C2C(C(N)=O)C2)=O)CC(F)(F)CC1CNC(=O)CC1CC(O)C12CCC2 c1(C2C(c3cn(C)nn3)C2)ccc(Br)cc1.c12ncc(s1)CC1CCN1C2=O.CO C1(NC(C(c2ccc(C)cc2)=O)=O)CN(C(=O)CC2CCCCO2)CCC1C c1(-c2c(C)nc(CC)s2)ccnc2ccc(C(=O)Nc3c(Cl)c(C)nn3C)cc12 C(=O)(CC1N(C(C2(O)CCCCCC2)=O)CCc2ccccc21)OC CC1(C)CCOC1CC(=O)NCC(C1CCC1)NC(c1c(F)cnn1C(F)F)=O C(C(=O)NC(C)(C)C)(C(C)CCC(=O)NC1CC1)N(CC(=C)C)C c1(OCCCC)ccc(C(=O)NCCC2CC(NC(=O)C(C)=C(C)CC)C2)cc1 O=C1CN(CC(=O)N(CCC2(O)CN(C(C3CC4CCC3C4)=O)C2)C2CC2)CCN1 Cc1oc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)NC1COC(C(C)C)C1 N1(C(C(CCCC)O)=O)CCCC12CCN(C(C13CCCC1(C(N)=O)C3)=O)CC2 C(CCCCC(=O)NCCC=O)NC(c1ccc(N)cn1)=O.C(N)(=O)O CC1CCC(C)(C(=O)NCC2(C(=O)NCC3(C#N)CCC3)CC23CCC3)CC1 C(CC(O)C(F)(F)F)NC(C#CCNC(c1n[nH]c(=N)[nH]1)=O)=O N1(C(CC=CC(C)(C)C)=O)Cc2n[nH]cc2C1C(=O)NC(C(N)=O)C1CCCC1 N(C1CCc2ccc3c(c21)CCO3)C(CCC1C(C)C1)C(=O)NC1(C)CC1 N1(C(c2c(OC)noc2C)=O)CCCc2ccc(NC(=O)C(C)N3CCC3)cc21 N1(c2nnc(C(C)F)n2CC2CC2)CCC(C2CC2)C1 C1(CCNC(c2occc2CO)=O)CCCCN1C(c1ccc(C(F)(F)F)[nH]1)=O c1(C(N2CC3CN(Cc4n[nH]cc4Cl)C3C2)=O)ccc2ccc(Cl)cc2n1 C(=O)(C(O)CC1CC1)N(CC(CN(C)C(C1CC(n2ccnn2)C1)=O)O)C N1(C(C2CCC(NC(c3ncc(C#C)cc3C)=O)C2)=O)CCC12CCCOCC2 C1(CC(=O)NCCN(C(COCC(c2ccccc2)C)=O)C)CCC(=O)N1 C=C=CCCC(=O)NCC1CC(NC(c2cccc(-c3ccoc3)c2)=O)CC1O C(=O)(C1=C(Cl)CCCC1)NC1CCN(C2CCN(C)C2=O)C1(C)C N1(C(C(C2CC2)SC)=O)CC(C)(CNC(c2cc3cc[nH]c3cn2)=O)CC1(C)C C=CCC(C)(CC=C)NC(=O)NCCc1nc(C)nc(O)c1C C12(C(=O)NCC3CC(CNC(CC(COC)C)=O)C3)CCCC1C2(F)F C(=O)(CCCC(=O)NCCCC1CN(C(=O)C(O)C(F)F)CCO1)NCC Cc1c(C(=O)NCC(C)NC(=O)C(O)Cn2cncn2)ccn1CCO Cc1ccc(C(C)(C)CC(=O)N2CCC(CCNC(=O)CCF)C2)cc1 c1(CN2CC(C(=O)Nc3ccccc3OC(F)F)SCC2)cc(F)cc(F)c1O c1(NC(c2ccc(NC(N3CCC(C(=O)OC)C3)=O)s2)=O)ccc(C)c(I)c1 c1(CN2CC(C)OC(c3ccsc3)C2)ccccc1[N+](=O)[O-] C(CCO)(C(C)(C)O)NC(c1cc(CNC(CCSC)=O)ncc1)=O N1(C(C2C(c3cn(C)nc3)C2)=O)CCN(C(=O)C=CC=Cc2cccnc2)CC1 n1(CC)ccc(C(=O)NC(CN(C)C(c2cnsc2)=O)(CO)CO)cc1=O C1(NC(c2n(C)cc(F)c2)=O)CN(C(c2ccccc2O)=O)CCC1(F)F C#CCC(C)(C)C(=O)N1CCC(CCCNC(c2cnn(CCC)c2Cl)=O)CC1 c1(C(N2CCOCC(NC(c3n(C)cc(Cl)c3)=O)C2)=O)nc2c(s1)COCC2 N1(C(=O)CN2CCOCC2)CCCC2CCN(C(C3(CC4CC4)CCC3)=O)CC12 CC1CCC(C)CN1C(=O)C(CC(F)F)NC(=O)C=Cc1cc[nH]c1 CCCC(O)CC(=O)NCC1CC(F)(CNC(C2(CF)CC2)=O)C1 CN1CCN(C(c2ccc(C(C)(F)F)nc2)=O)C(CNC(c2csc(Cl)c2)=O)C1 C1(C#CC(=O)N2CCC2C2CN(C(C3CCCCS3)=O)C2)(CC)CC1 c1(CNC(C(C)OCC)=O)ccc(C(N2CCCC2(C)CO)=O)cc1 Cc1c(C(=O)OC(C)C)cccc1[N+](=O)[O-].c12ccnc(c1)NC2 c1(C(=O)NC2C(CC)CN(C(=O)C(F)CC3CCC3)C2)csc2cncn12 c1(C(=O)NC2C(NC(CC=CCC)=O)COCC2)cccc2c1NCCC2 N1(C(CS(CC)=O)=O)C2CCC1C(C(=O)NCC1C3CCCCC13)C2 Cn1cc(C#CCNC(C2CCN(S(=O)(=O)C(F)F)CC2)=O)cn1 CC(CCCc1ccccc1)C(=O)NCCOCCCNC(=O)CCCN(C)C c1(C(=O)NC2CN(C(c3cnc(C)[nH]3)=O)C2)ccc(Br)c(C)c1F C(c1ccc2ccccc2c1)=C(C#N)C(=O)NC1CC1NC(c1ccoc1Cl)=O C1(CC(N)=O)(NC(c2cccn2CCC)=O)CCN(CC(=C)Br)CC1 C1(NC(C(C)(C2CC2)OC)=O)CCCN(C(=O)Cn2ccnn2)C1 C(C)(c1ccncc1)=CC(=O)NC1OCCN(CC)C1 C(=O)(CCCF)N(C(C(=O)NC(C1CCOC1)C#C)C)C C1(C(=O)NCC2CCC(C(=O)NCCCNC(=O)OC)C2)CC(F)CN1C CN1C(=O)CCCC1C(=O)NC1CCN(C(C2(c3ccccn3)CC2)=O)CC1 c1(C(N2CC=CC(NC(C3ON=C(CC)C3)=O)C2)=O)cn(C)c2ccc(Cl)cc12 N1(C(C=CCCC)=O)CCC2(CC2)CC1C(=O)Nc1cc(O)ccc1C CC1=CCN(C(C2(C3CCCN3C(=O)Cn3cccc3)CC2)=O)CC1 CCC(CC(C)C)C(=O)NC1CC12CC(NC(c1nn(C)cc1Cl)=O)C2 CC1CC(C(=O)N(C2(C(=O)NC(C)(C)C)CC2)C)=NO1.C1(=O)C(O)CCN1 Cc1cc(C)c(C(=O)NCCN(CC(C)O)C(=O)COCC(C)(C)C)s1 CC(CNC(=O)CC12CCCC1C2)(CO)NC(=O)CSc1nnc(S)s1 C(CC)(C(=O)N1CC=CC1C(=O)NCCC(=O)NC(C)C)OCC.OCC C1(COC)CN(C(c2cccnc2N)=O)CCN1C(=O)C=CC1CCOC1 C1(NC(C(CO)OC)=O)CN(C(=O)COc2cccc(F)c2F)CC2CCCC12 CCC(CC(F)(F)F)C(=O)N1CC(NC(=O)C=C2CCN(C)C2)C(C(F)F)C1 Cc1cc(C(=O)NC2CCC(NC(=O)Cc3c(C)noc3Cl)CC2)nc(O)n1 C12CC(C1)NC2=O.C1(C(=O)N(C)CC2(CC(C)C)CC2)(CC)CC1 C1(NC(CC2CC(=C)C2)=O)CC(c2ccccc2)(NC(=O)Cc2coc(C)n2)C1 c1(C(=O)NCC2N(C(c3c(Cl)cnc(C(C)C)n3)=O)CC2)cccc2[nH]ccc12 C1(NC(c2c(C)nncc2)=O)CC2CC(C1)N(C(=O)CN(C)C(N)=O)C2 C12CC13CCN(CC3)C(=O)NC2.CCC(CC)C(C)OC.C(C)(C)(C)O C1(NC(=O)NCCCCC2C(C)C2)CCN(C(=O)C2(C#N)CC2C)O1 Cc1ccc(NC(C2(C)CCN(C(C3CCCN3C)=O)C2)=O)c(O)n1 C1(NC(C2CCC(C)O2)=O)CC2CN(C(c3coc(Br)n3)=O)CCN2C1=O N1(C(=O)CN2CCCCC2)CCC(C2CCCN2C(C2CCCOCC2)=O)CC1 C(C(C(F)(F)F)N1CCNCC1)NC(c1sccc1C(=O)Nc1ccccn1)=O C1(CC)CNC(=O)CN1C(=O)C(C1CC1)NC(c1cn(CCO)nn1)=O Cc1ccc(C(=O)N(C)CCOCCNC(C2C(c3ccccc3F)C2C)=O)nn1 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC2(CCC2NC(C2CCCCS2)=O)CC1 CC(C)CC(C)(CNC(=O)CC1CCN(C)C1)NC(C1CC(C)(F)C1)=O c1(-n2c(-c3c(C(C)OC)nn(C)c3)nc(CO)n2)ccc(C)cc1C CC(O)(CNC(c1cc(Br)c(Cl)s1)=O)CC(=O)O N1(C(CC2CCCN(C(C(CCCC)N(C)C)=O)C2)=O)CCC(F)(F)C(F)C1 O=S(=O)(c1ccc(CC23COC(CF)(C2)C3)c(Cl)c1)NCC1CCN(CCF)C1 C(=O)(CC(O)CN(C)C)NCC(CC)NC(=O)C(c1ccc(OC)cc1)(C)C C(=O)(C(Cc1ccccc1)CC)NC(CNC(CN(C(CC)(C)C)C1CC1)=O)CO CC(CS(C)=O)C(=O)N1CCC(=CCNC(c2nnn(C(C)(C)C)n2)=O)CC1 c1(C(=O)NC(C)CCNC(=O)CSC(C)(C)C)cc2c(nc1O)C(C)(C)CCC2 C1(c2ccc(C)nc2Cl)CC2(C1)NC(=O)N(CCC1CCCCO1)C2=O C(CN=c1ccnc(NCC(N)=O)[nH]1)(C(C)(C)C)N(CC)CC C(CC)(CC(CC)CC)NC(C1CCN(C(C(CC#C)O)=O)C1)=O c1(CCNC(C2C(CNC(C=C(C)C(C)C)=O)CCC2)=O)cc(C)n(C)n1 C1(CNC(C=C(C)C(F)F)=O)(CNC(C2(C#N)CCCO2)=O)CCOCC1 c1(C(N2CCC(CNC(=O)C(F)(Cl)c3ccccc3)C2)=O)nccc2occc12 CC1CC(C(=O)NCC2(CCNC(=O)CC3C(C)(C)C3(C)C)CC2)CC(C)(C)C1 c1(OCC)ccc([N+](=O)[O-])c(NC2CC(C)N(C(=O)C(c3ccccc3)F)C2)n1 C(=O)(C(CN=[N+]=[N-])NC(c1ccc(C)cc1)=O)NCc1c(CC)nn[nH]1 CN1CCCC1CC(=O)NCC1CC(NC(c2cn(C)nn2)=O)C1 c1(CC)nc(C)oc1C(=O)N(CCCN(C(=O)C=CC1CCCN1C)C)C c1(C(C)NC(C(=O)OC)(C)Cc2ccccn2)cccc(Cl)c1C Cc1nc2c(s1)CC(C(=O)NC(C)(C)CNC(=O)COCCCF)CC2 C1(C(N(C2CC2)CC)=O)CC(O)(CNC(=O)COC2CCC2)C1.C1CC1 C(=O)(C1=CC(O)C(NC(C23CCC(CC2)C3)=O)C1)NCCC1(C)CCCC1 C1(CCCC)CN(C(=O)CSC)CCN1C(=O)CC(F)F.c1(CCC)ncc[nH]1 Cc1ccc2c(C(=O)NC(C)(C)CN(C)C(c3nnn(C)c3N)=O)ccnc2c1 C12(C(=O)N(C3(C)CCC(C)C3I)CC)COC(=O)N1CCN(C(=O)OC(C)(C)C)C2 CC1C(C)N(C(C2SCCS2)=O)CCN1C(=O)CCCS(C)(=O)=O CC(C)C(CN(C)C)C(=O)NCC(C)N(C)C(c1ccccc1N1CCCC1)=O CC1CCCN(C(=O)C2=CCSC2)C1CNC(=O)CCOc1ccc(F)cc1Cl c1(OC)cc(F)ccc1C(N1CCC(O)(CC#N)C1)C(=O)NC(C)(C)C N1(C(c2cc(C)on2)=O)CCCC(NC(=O)COC(C)C)CC1 O=C1CCC(=O)N1C1CCCC1CSCOCc1cncnc1 C1(C(=O)NCCCS)CC2CC1C1CC21.C1(NC(C2C(C)(Br)C2)=O)CCN(C=O)CC1 O=S(=O)(c1ccc(CO)c(Cl)c1)N1CCOC(c2ccc(C(F)(F)F)cc2)C1 C1(CNC(COC)=O)CCN(C(=O)COc2cnn(C)c2)CCC1(F)F N1(C(C(C)(C)CO)=O)CCC2(CCC2NC(C23C4CCC(CC24)C3(F)F)=O)CC1 C1(C(=O)NCC(C)OCCO)CC2(CCN(C(=O)C(c3cccnc3)O)C2)C1 C(=O)(CCCS(C)(=O)=O)NCC1(CNC(c2n(C)c(S)nc2)=O)CCCC1 c1(C(=O)NC(CCN(C(CC=CCC)=O)C)C(C)C)cnn2c1OCC(OC)C2 c1(CN(C)C(C2C=C2C)=O)nc(CC2CN(CCOC)C2)co1 N1(C(=O)NCC(=O)NCc2ccc(C)cc2)CCCCc2cc([N+](=O)[O-])ccc21 C1(CNC(C=C(C)Cl)=O)CCCCN1C(=O)CNC(c1ccc(N)cc1)=O c1(C(=O)NCC2(CNC(C(C)NC(=O)NC)=O)CCC2)ncn2ccc(C)cc12 NS(=O)(=O)C1COc2c(C(=O)Nc3cc(Cl)cc(Cl)c3Cl)cccc21 C1(CC(=O)NCCNC(c2[nH]ccc2-c2ccccc2)=O)CC2C=CC1C2 c1(OCCCC)ccc(CCN(C(C2CC(n3ccnn3)C2)=O)C2CC2)cc1 c1(CSCCOC(CS(CC)(=O)=O)=O)sc(S(N)(=O)=O)cc1C.C12CCCCN1C2=O C1(NC(=O)Cc2ncc(Cl)s2)CC(CNC(=O)Cn2cc(C3CC3)nn2)CC1O C1(C(=O)NC2CC(CNC(CNC(=O)OC)=O)C2)CC2(COC(=O)N2)C1 C(CC(C)(C)CNC(c1ccc(NC=O)cc1)=O)NC(Cn1c(C)cnc1)=O N1(C(C(CCC)N(C)C)=O)C2CCC1CN(C(C1C3COCC13)=O)C2 C12(OC(C)(C)C)CC(NC(=O)C(N3CCC(CC4CCOC4)CC3)=O)(CCO1)C2 C(=O)(C(CNC(C1(OC(C)C)CC1)=O)CC1CC1)NC(CC)(C)C(N)=O N1(C(c2cn(CC)nc2)=O)CCCCC1C(=O)NCCCOC1CC1 c1(C(=O)NCC(CC)NC(c2cccc(C(C)C)n2)=O)ccc(C2(C)CC2)cc1 N1(C(C(CC)N(C)C)=O)CCOC2CCN(C(=O)C=C(C)c3cnn(C)c3)CC12 S(=O)(=O)(c1csc(C(N2CCCC(NC(c3cnc(N)c(Cl)c3)=O)C2)=O)c1)NC CN1CCOC(C(=O)NC2C3CC(NC(C4(CO)CCOCC4)=O)CC23)C1 C1(CC)CN(C(=O)CO)CCC1CNC(=O)C(c1ccc(Br)c(F)c1)C C(=O)(C(C)(C)NC(=O)C(F)(F)F)N(C1CN(c2nnnn2C)C1)C N1(C(C2N(CC(C)C)CCC2)=O)CC2(NC(c3cc(C(C)(C)C)no3)=O)CC1C2 C1(CC(=O)NC2CC(CC)C2)CCN(C(=O)C(C)S(N)(=O)=O)C1(C)C Cc1cc(Cl)ncc1NC(C1CCCN(C(=O)C(c2ccc(F)c(F)c2)O)C1)=O CC1COC(C(=O)O)CN1C(C1CCN(C(=O)Cc2cncnc2O)CC1)=O c1(CCCNC(=O)NCC2(c3ccc(F)cc3)CCCCC2)ccc(O)c(O)c1 c1(CC2(C(=O)NCCN(C(C3CCCCS3)=O)CC)CCC2)ccc(F)c(F)c1 c1(OCC)cc(Cl)ccc1NC(N1CCNCCC1C)=O c1(NC(C2(F)CCCN(C(C(C)Cn3ccnc3)=O)C2)=O)ccc2c(c1)OCC2 c1(C(=O)OC)ccnc(N2CCN(C)CC2CNC(=O)C=CC2CC2)c1[N+](=O)[O-] CCCCC(C)C(=O)N1CC2(CC)CC1(C(=O)N(C(CC)C1CC1)CC)C2 C1(CC)(NC(=O)C2CC2)CCN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC1 C(C(=O)NCc1ncc(C)[nH]1)(C(C)CC)N(C(CCC=C=C)=O)C N1(C(c2ccon2)=O)CCC(C2(O)CN(C(C3CCCS3)=O)C2)CC1 CC(C)P(=O)(CC(=O)NCC(C)(C)NC(=O)CCc1ncccn1)C(C)C c1(C(=O)NCC2CCC(NC(CCN(CCC)C)=O)C2)ccc(Cl)c(N)c1 CCCCCCC(CC)C(=O)N1CCN2CC(NC(=O)CCC3CC3)CC2C1 C(C1=NOC2CCCCC12)n1cc(Cc2n(CC)ccn2)nn1.C1C(C)CC(=O)N1 c1(NC(C2(C)N(C(CNC(C)=O)=O)CC2)=O)c([N+](=O)[O-])cc(Br)cc1[N+](=O)[O-] CC(C)C(CNC(=O)CCCNc1ccccc1Cl)C(=O)O C(CCCC(C)(C)C(=O)NNC(=O)C(O)C1CC1)NC(C1ON=C(CC)C1)=O C1(CC)C(NC(=O)COCCOC)CCCN1C(=O)CC1CC(=O)NC1=O N1(C(c2c(CC)n[nH]c2)=O)CCC2CC2(C(=O)NC2CCN(C)C(=O)C2)CC1 CON(CCC(=O)OC(=O)C(C)CSC)C(=O)C1=CC(C)(C)C1 C1(CNC(c2c(OC)nn(C)c2)=O)C2CCC(C2)N1C(c1ccc(C(N)=O)o1)=O c1(C(=O)NC2C(NC(C3CC(=O)NC3)=O)C2)cc2ccccc2s1 Cc1c(C(=O)NC2CC(C)N(C(=O)CC3CCC(=O)NC3)C2)cnn1C(C)C CC(CN(C)C)CC(=O)N1CC(O)(C(F)C(=O)N(C)CCC2CCCCC2)C1 C1(CC)CCCN(C(=O)CCC(C)OC)C1C(=O)NC1CC(CO)C2CC12 N1(CC)CC(C)(C)OC(=O)C1CC(=O)NCC(CC(C)C)NC(C1CCSC1)=O C(=O)(C(C)(C)C(=O)N(C)C)NCC(C)CNC(c1cncn1C1CC1)=O CC1CC2CN(C(=O)CC3CCOCC3)CC2N1C(=O)Cc1cccc(Br)c1 CC(C)C(N=[N+]=[N-])C(=O)NC1CC(C(=O)NCCOc2ccncc2)CC1O N1(C(COC2CN(C(C3(OCC)CCC3)=O)C2)=O)CC(C)OC2(CCC2)C1 C(C)(C)(CC(=O)NC(C(O)CO)C1CC1)N(C(C1(CC#C)CCC1)=O)C C(=O)(C(F)C(C)CNC(c1cscc1Cl)=O)N1CC(COCC)C1 c1(C(=O)NC(C2CCN(C(C(CC=C)C)=O)C2)(C)C)noc2ncccc12 C#Cc1cccc(C(=O)NC2CCC(NC(=O)CCc3ccncc3)CC2)c1F Cc1cc(C(=O)NCC=CCNC(=O)C(C)(C)c2ccn(C)n2)cnc1C c1(C(=O)NC(CNC(c2cn(CCC)nn2)=O)C2CC2)cn(C2CCC2)nc1C c1(C(=O)Nc2ccc(N(Cc3ccc(C)s3)C3CC3)c(F)c2)cc(F)c(F)c(F)c1F c1(C(=O)NC2(C)CCN(C(=O)CC3CCCCO3)C2)nnc2n1CCCC2 c1(C(=O)NC(C)CNC(C2(c3ccccc3)CCOC2)=O)cc(C(N)=O)cn1C c1(C(=O)NCC2(C(N3CCCC(F)CC3)=O)CC(=C)C2)ccnc(C)c1C C1(CNC(C(C=C)CC)=O)CN(C(c2cnsc2C)=O)CC1(C)C c1(C(=O)NCC(C)N(C(c2ccc(NC)cn2)=O)C)cn(C)ccc1=O N1(C(c2cc(COC)on2)=O)CCN(C(=O)Cn2nc(C)cc2C)C(C)C1 CC1(C)COCC(CC(N2CCC(C)(NC(c3cncc(N(C)C)c3)=O)C2)=O)O1 c1(C(N(CC(C)NC(c2cc(-c3ccccc3)co2)=O)C)=O)csc(Cl)n1 C(=O)(CC(C)CF)NCC(C)CN(C(=O)CCc1ccc(Cl)cc1)C N1(C(C2(OC)CC2)=O)CCC(CNC(c2ncccc2CN(C)C)=O)C(F)(F)C1 CC1C(=O)NCCN1C(C1CCC(C)CN1C(c1ncnc(O)c1F)=O)=O N1(C(c2ccc(NC(N)=O)cc2)=O)CCCC(C)C1CNC(C1C(OC)C1)=O C1(C(=O)NCC(C)(CSC)NC(Cc2c(CC)con2)=O)(C(N)=O)CC(F)(F)C1 N1(C(C2CC(C)(C)C2)=O)CCCC(C)(C)C1C(N1CCC(CCF)CC1)=O CON(CCC(=O)NC1CC2CC3C(C2)C13)C(=O)c1cccc(C)c1 C1(NC(C2=CC(C)(C)C2)=O)COC2(CCN(C(c3csnc3Br)=O)C2)C1 c1(CC(=O)NCC(C2N(C(CC(C)(F)F)=O)CCCC2)(C)C)ccc(F)c(F)c1 N1(C(C(C=C)(C)C)=O)CCC2(CCCN(C(c3nnc4ccccn34)=O)C2)CC1 C1(CNC(C(C(=C)C)(C)C)=O)COC(C)(C)CN1C(=O)C(C)CC(C)C c1(C(=O)NC2(C3CN(C(C(C)SC)=O)C3)CC2)nc(Br)n2ccsc12 N1(C(c2c(C)ncs2)=O)CC2CCCC(C1)N(C(=O)Cn1ccc(Br)n1)C2 C1(C(N(CC)CC2CCN(C(C3CC3C)=O)CC2)=O)Cc2ccccc2S1 C1(CN(C)C(c2cnc[nH]2)=O)CN(C(=O)Cc2cccc(O)c2)CC12CC2 C1(n2ncc(NC(=O)Nc3cnc(C(C)C)n3C)c2)CCC2(CCC2)CC1 Cc1ccc(C(N2CC(CNC(=O)COC(C)C)OC(C(F)(F)F)C2)=O)c(O)n1 c1(OCC)cccnc1N(C)C.c1(C(c2nnnn2C(C)C)N)csc(C(F)F)c1 n1(CC(=O)N(C2CCN(C(c3c(CC)[nH]nc3Cl)=O)C2)CC)ncc(O)nc1=O C12(C(=O)NCCN(CC(C)O)C(c3ccon3)=O)CC1COC2(C)C C(CCC)(CCC)=CC(=O)N(C(C)C(=O)NC(C)CCCC)CC#C N1(C(CN2CC(C)(C)C2)=O)CCC=CC1C(=O)NCc1cccnc1 N1(C(CC2CC(SCC)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)C2CC12 N1(C(C2(C#N)CCCO2)=O)CCCC2(CCN(c3ncnc4[nH]ccc34)CC2)C1 C1(NC(C2CC3CCC2C32CC2)=O)CCCC12CCN(C(=O)CCF)C2 C1(NC(C2CN3CCCN2CC3)=O)CCSC12CN(C(c1cnns1)=O)C2 c1(OCC)cc(C)ccc1C(=O)NCC1(Nc2nccc(C#N)n2)COC1 S(=O)(=O)(c1ccc(Br)cc1)NC(C(CCCC)NC(=O)CN)=O Cc1sc(O)nc1C(=O)NC(C(C)NC(c1ncccc1F)=O)C(C)C C1(C)(C(=O)OCC)CCN1C(C1CCC(NC(=O)CNC(=O)CC(C)C)C1)=O C1(OCCC)CCCN(C(C2CC2c2nnn(-c3nc(C)c(Br)s3)n2)=O)CC1 C(C1Cc2ccccc21)NC(C1N(C(C(COC)(C)C)=O)CC(F)C1)=O c1(C(=O)NC(CNC(c2c(CC)scc2)=O)(C)CO)ccc(OCCF)cc1 C(=O)(C1=CCCOCC1)NC(C1CCCC1)CNC(c1c(C)nn(C)c1C)=O N1(C(CC2CC(C)C2)=O)CC=CC1(C)C(=O)NC1(C)CCC1 C#CCC(C)C(=O)NC(C)CC(C)NC(C12CC(C1)C(C(F)(F)F)O2)=O c1(C(N2CCN(CC(C)O)C(CCO)C2)C(=O)NCC=C)cc(Cl)c(Br)c(Cl)c1 c1(C(N2CCC(F)(CO)C2)C)ccc2cc[nH]c2c1.C1(=O)CCCN1 C1(CNC(C2N(C(C(C)C)=O)CSC2)=O)CCC2(CC1)CC2 c1(C(C)C(N2CCC(N(C(=O)COCCF)C)C2)=O)ccc(Br)cc1F CC1CN(C(=O)Cc2cccc(Cl)c2)CCC1N(C(=O)CCn1ccnc1)C Cc1cc(C(=O)NCC2CC(O)CN2C(c2cnn(C)c2)=O)nn1C(C)C1CC1 C(=O)(CC1CNc2ccccc21)N1C(CNC(C2CCC3C(C2)C3(F)F)=O)CC1 CC1CN(C(C2(O)CCOCC2)=O)CCN1C(C1CN(C2CCOCC2)C1)=O c1(OC)ccc(NC(=O)CCC(=O)N2CCC(NC(=O)C(C)C(C)C)C2)c(C)c1 N1(C(COC2C(CC)CCC2)=O)CCSCC1CCNC(=O)COC(F)(F)F N1(C(C2CC(C)(O)C2)=O)CC2CC1C2CNC(c1ncccc1C(F)(F)F)=O c1(C(=O)NC(CN(C(C2C(OC)C2)=O)C)(C)C)cc(C)c2ncccc2c1C CC1C(C(F)(F)F)OCCN1C(=O)NCCC1CCOC(C)(C)C1 C12(C(N3CC(C#C)(N(C)C)C3)=O)CC(CCO1)N(C(c1cc3ccccn3c1)=O)C2 c1(CSCC2CC(OC(C)C)C2)cccnc1O C1(C(=O)NC(C(C)C)C2CCC2)CCOCCN1C(C1CC(C)(F)C1)=O C1(CC(C(N)=O)CNC(C2CCCC(=O)C2)=O)CCC(F)(F)CC1 Cc1nnc(CCC(=O)NC(C2CCN(C(=O)C(C)n3ccnc3)C2)(C)C)o1 C1(OC(C)C)CCN(C(C2CN(C(C3CC3(F)Cl)=O)CC2C(C)C)=O)CC1 N1(C(C(C)OCCOCC)=O)CCCC(C)(CNC(=O)CCCN2CCCC2)C1 c1(CNCC(C(=O)N(c2cccc(-c3cnnnc3)c2)C)(C)C)cn(C)nc1Cl N1(C(c2nc(CC)oc2)=O)CCCOC(CNC(c2ccnc(Cl)c2Cl)=O)C1 C1(NC(=O)NCC2CN(C)C(=O)C2)CC2(CCN(C(C3(CSC)CC3)=O)CC2)C1 C1(CNC(C=C(COC)C)=O)CC(C)CN(C(C2CC(C(=O)OC)C2)=O)C1 c1(CCNC(c2cc(N3CC(CCOC)(C(=O)OC)C3)sn2)=O)ccc(C)c(C)c1 C(=O)(CCCS(C)(=O)=O)NC(C1N(C(c2n(CCC)ncc2Cl)=O)CCC1)C C1(NC(c2c(C)nccn2)=O)CN(C(=O)Cc2cnoc2)Cc2ccnn2C1 O=C(CCCCCBr)N1CCN(C(c2cnn(-c3ccc(Cl)cc3)c2)=O)C(CO)C1 c1(SC)ccccc1C(F)(F)C(=O)N(C(CNC(C1(n2ccnn2)CC1)=O)C)C C(=O)(C(C)C(C)(C)C)NC1C(C(=O)OC)CN(C(=O)C(F)=C(C)C2CC2)C1 C12(CC(N3CC(C(=O)NC45CCC(OC)C4C5)OCC3)=O)CC3CC(CC(C3)C1)C2 CC(N=c1[nH]c2ccc(Br)cc2s1)C1CN(C(C2CC(C)(F)C2)=O)CCO1 N1(CCN(CC)CC)CCN(C(C2(C)CCN(C(=O)C(=O)C3CC3)C2)=O)CC1 N1(C(C)Cc2ccccc2Cl)CCC2(CC1)CC2C(=O)NC(C)CCO Cc1n[nH]c(C)c1CC(C)C(=O)N(CCNC(C1(O)CC(C)(C)C1)=O)C1CC1 CC(C)(C)C(CNC(C1(C#N)CCCC1)=O)C(=O)Nc1cc(C#N)ccc1O C(C(=O)NC(C1(O)CN(C(=O)CC(C)(C)C#N)C1)C)(C(C)(C)C)SC C(CN=c1cc(C(C)(C)C)nc[nH]1)(C(C)(C)C)NC(C(CC(C)(C)C)O)=O n1(CC)nc(C)c(CC(=O)NCC(O)CN(C)C(c2ccn(C3CC3)n2)=O)c1C N1(C(C(C)N(C)C)=O)CCC(N(CCO)C(c2cc(C3CC3)ccn2)=O)CC1 C1(NC(C2N(C(C(CC=C)CC)=O)CCC(=C)C2)=O)CCC2CC1C2(C)C c1(OC)ccc(C(=O)NC2COCC2NC(C2(CO)CC2)=O)c(F)c1Cl C1(N(C(c2csc(C3OCCO3)c2)C(=O)NCC(=C)C)C)CCCCC1C C(CO)(CC(O)c1ccccc1)N(CCNC(C(C)C)=O)CCC N1(C(C2S(=O)(=O)CC(N)C2c2ccccc2)=O)CC2(CCOCC2)CC1CO N1(C(C2C(C)C2C)=O)CC(NC(=O)COCc2ncnn2C)CC(O)C1 C(CN=c1[nH]c(=NCc2ncsn2)[nH]c2c1CSC2)n1cc(Cl)nn1 C(=O)(C1=C2CCCN=C2NN1)N1CC(NC(c2cc(C)nc(C)c2)=O)C(C)(C)C1 c1(N2CCC(F)(CN(C)C)C2)nc(=NC2C3CCCOC23)[nH]c2c1SCC2 C1(C(N(C2CCC(N(C)C)CC2)C)=O)=NC=CC(C(F)(F)F)=NN1CC1CC1 c1(C(N(CCN(C(=O)C=CC(N2CCOCC2)=O)CC)CC)=O)cnnc(C)c1 Cc1cc(C(N2CCC(C)(CNC(=O)C(F)C(C)(F)F)CC2)=O)c(C)cn1 C(=O)(C(C)(C)CCC)NC(CC=C)C(=O)NCC1(O)CC2C=CC1C2 N1(Cc2c(NC(c3cccc(F)c3O)=O)cccc2)CCC2CN(CC)CCC12 C(C(C(C)C(C)C)NC(=O)CSCCC#N)NC(CCCOCC)=O c1(OC)cc(C(=O)NC2CC(CNC(c3ccn(C)n3)=O)C2(C)C)cc(F)c1 c1(OC)cnccc1-c1nc(C)c(NC(c2scnc2C(F)(F)F)=O)s1 c1(C(=O)NC2CN(C(C(C)SCC)=O)CC2SC)c(C2CC2)cccc1F C1(CNC(c2c(OC)nsc2)=O)CC2(CCC2)CN1C(c1cc(CCO)on1)=O c1(C(N2CCCC(NC(CCC=C)=O)C2)=O)cnc(C(F)(F)F)c(F)c1 N1(C(c2[nH]cc(CC(C)C)c2)=O)CCCC(CO)(NC(c2ccn(C(F)F)n2)=O)C1 C1(F)(C(N2CCC(CNC(c3c(C(C)C)nn(C)c3)=O)C2)=O)CC12CCCCC2 N1(C(c2c(C)cncc2)=O)CCC2(CC1)CCN(C(=O)COCC1CC1)C2 c1(NC(C2CC(NC(c3c(C)n[nH]c3C)=O)C2)=O)c(F)c(F)nc(F)c1F CCC(CC(=O)NC(C1CCCN(C(c2cncc(OC)n2)=O)C1)C)CC(C)C c1(-c2cn(CC(CC)O)nn2)ccc(C(N(CCN(C)C)CC)=O)cc1 N1(C(c2cc(C)nc(C)n2)=O)CC(C)(C)OCC1CNC(c1cc(C)sn1)=O C1(CNC(C2CC(N(C)C(c3cscc3C(F)F)=O)C2)=O)CN(C)CCN(C)C1 CC1(CCNC(C2(C)COCCO2)=O)CCN(C(=O)CCC2CC(F)(F)C2)C1 CCCC1C(=O)N1.c1(CNC(=O)OC(C)(C)C)ccc(OCC(F)F)nc1 N1(C(C2(CC=C)CC2)=O)CCC(CNC(=O)CCc2cn(C)nn2)(COC)C1 Cc1ccc2c(N(C(=O)C(=O)NCC3CCCN3C(=O)C(C)(C)C)C)c[nH]c2c1 CCC(CC(F)(F)F)C(=O)NC1C(CO)N(C(c2cn(C(C)C)nn2)=O)C1 N1(C(CC)=O)CCC(F)(CNC(=O)C2=CCCOC2)CC1 c1(C(N2CCC(CCNC(C3C=C(C)CS3)=O)CC2)=O)ccnc2ccsc12 C1(NC(=O)CC2CC3(CCC3)C2)CC2CCC(C1)N2C(=O)Cc1ccco1 C(C(C)(C)CO)(c1ccccc1)NC(=O)NC(c1ccc(C)o1)CC Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C)(O)CNC(=O)C(C)(C)CO CC1CN(C(c2ccon2)=O)C(C)CN1C(=O)CC1(N(C)C)COC1 Cc1nc(NC2CCCC(NC(=O)C=CCF)C2)c2cnn(C)c2n1 C(=O)(CCCCCCNC(c1nonc1N)=O)NC1C(CC=C)COC1 c1(CNC(=O)OC(C)(C)C)cncc(N2CCCC2)n1.C(=O)(CS(C)(=O)=O)N c1(C(N(C)CC2(OCC3C(C)C3)CC2)=O)cnc(S)n1-c1ccccc1.C1C(=O)N1 c1(NC(C2C(C(C)C)N(C(=O)COc3ccccc3)CC2)=O)cc([N+](=O)[O-])sn1 CCCC(CC(=O)NCC(C)(C)C(C)C)NC(=O)C(O)CC1CCCC1 c1(C(N)=O)ccc(C(N2CC3CC2C3CNC(C2CCNC2=O)=O)=O)nc1 C#Cc1cccc(C(=O)NCC23CCC2CCN3C(c2n[nH]c(C)c2C)=O)c1F c1(NCC2(OC)CC(C(C3CC3C(=O)N)=O)C2)c(C)noc1C.C(=O)(OC)NC1CC1 N1(C(c2c(C)cc[nH]2)=O)CCc2ccc(C(N3C4CSCC3C4)=O)nc2C1 C#Cc1ccc(C(N2CCC(CNC(=O)C=Cc3cncs3)CC2C)=O)cc1 c1(C(CNC(C2(COC)CC2)=O)NC(=O)C(=Cc2cccs2)C)ccc(F)cc1 Cc1ccc(N2CCC(N3CCCC3(C)CN)C2=O)cc1 N1(C(c2cnc(CNC(C3N(C)CCC3)=O)nc2)=O)CCCC(C2(C)CC2)C1 C1(C(=O)NC2CCC(N(C(c3c(CC)nns3)=O)C)C2)CC2C=CC1CCC2 C1(CC=C)(NC(c2cnn(CCO)c2C)=O)CCN(C(c2ccc(C)n2C)=O)C1 C1(C(=O)NCC2(OC)CN(C(=O)C(C)(O)c3ccccn3)C2)CC(=O)OC1(C)C C1(C(N2CC(C(N)=O)(CNC(C(COC)C)=O)C2)=O)(CO)CCCCO1 N1(C(C2CCN(C(c3c(NC)nccc3)=O)C23CC3)=O)C2CCC1CC(F)C2 N1(C(C(CNC(c2oc(C)c(CO)c2)=O)CC2CC2)=O)CC(F)(F)C(F)(F)C1 c1(NC(=O)Nc2ccc(N3CCNCC3)cc2)ccnc(Br)c1F n1(C(CNC(c2nnnn2CC)CCC)C)cc(Br)cn1 C(=O)(CC(C)NC(N)=O)NC1C(C(=O)NC(c2nc[nH]n2)CC)CC1 N1(C(c2c(CC)n(C)nc2)=O)C(C)C2CC1C2NC(c1cncnc1C)=O N1(C(CNC=O)=O)CC2(CNC(c3cccc4oc(Cl)cc34)=O)CC(F)(C1)C2 c1(C(=O)NC2CCN(C(=O)C3=C(Cl)CCC3)C2C2CC2)cc2c(F)cccc2s1 C(=O)(CCCCCC(C)C)N1CC(NC(=O)CN2CC3CCC2C3)CC(OC)C1 C(N=c1[nH]c2ccc(O)cc2s1)C1CN(Cc2c(C(=O)OC)ccs2)C1 c1(C(c2cccc(F)c2)NC(c2cn(C)nn2)CC)cccc(Br)c1 C1(C(N2CCN(C(C(CC)CC)=O)CC2)=O)CCc2nc(C)ncc2C1 Cc1ncnc(O)c1CCC(N1CCCC(NC(C2(C#N)CC23CCC3)=O)C1)=O N1(C(C2(C=C)CCC2)=O)CCCOC(CNC(=O)COc2ccc(F)cc2)C1 c1(C(N2CC(CNC(C3=NOC(C)C3)=O)C2)=O)cccc2c1nc(O)n2C N1(C(C(CC)CC)=O)CCCOC(CCNC(=O)CN(C)S(N)(=O)=O)C1 c1(C(N2CCCS(=O)(=O)CC2)=O)cnn2c(F)cccc12 c1(C(=O)Nc2ccc(NC(C3CC3(F)F)=O)cc2F)cccc2cccnc12 c1(C(N2CC=CC(NC(C(C)OC)=O)C2)=O)cnc2c(c1)N(C)CCO2 c1(C(=O)NCCCNC(c2ccc(CC)o2)=O)ccc(N(C)C(C)C)cc1 N1(C(C=C(C)C(F)F)=O)CCC2C(CCCN2C(=O)Cc2cccc(Cl)c2)C1 C(c1ccc(O)cc1)=CC(=O)NCC(c1ccccc1)NC(c1n[nH]cc1Cl)=O C(CCNC(C1CCCCS1)=O)(C(=O)NOC1CCCC1)OC c1(C(N2C3CCC(NC(CCS(C)=O)=O)(C3)C2)=O)ccnc2cc(Cl)ccc12 C(N=c1cc(C)c(S(=O)(=O)N2CCCC(C)CC2)c[nH]1)C1(OCC)CCSCC1 Cc1oc2ccccc2c1C(C)N(C(N1CCC(O)C1c1ccccc1)=O)CCN Cc1ccc2cc(C(N3CC(NC(C4CCCC4(C)C)=O)C(O)C3)=O)ccc2c1 c1(C(N2C(CCOC)CN(C(C3CCC(O)C3)=O)CC2)=O)sc2cncn2c1C C1(C2CCN(C(C3CCC(F)CC3)=O)CC2)(NC(c2cnn3c2CCC3)=O)CC1 CN1CCCC(C(N2CCCC2C(=O)Nc2ccccc2CC(=O)O)=O)C1 C(C)(c1cccc(Cl)c1)=CC(N1CC2(CC(CNC(C=CC)=O)C2)C1)=O Cc1nc(C(=O)NCC2(F)CN(C(C3CCC=CCC3)=O)C2)nn1C CC1CC(C(=O)NC23CC(C2)N(C(=O)CCc2ccncn2)C3)CCS1(=O)=O C12(C(=O)NCCC(C)N(C)C(c3nonc3N)=O)CCCC1C2(F)F c1(C(=O)NCC(C)CN(C)C)ccc(NC(C2(O)CCCC2)=O)nc1.C(C=CCO)N C(=O)(CCCCCCCCNC(C)=O)NC1C2CC(OC)C(CC2)C1 c1(C(=O)NCC2C(NC(CCCC)=O)CCC2)cc2cccc([N+](=O)[O-])c2[nH]1 Cc1c(Cl)ccnc1C(=O)NC12CCC(CNC(=O)C(C)NC=O)(CC1)C2 C=CC(F)(F)C(=O)N(C)CC1CC(F)CN1C(=O)CCCc1cccs1 c1(CNC(C=CC(C)SC2CCN2C(=O)OC(C)(C)C)=O)ccc([N+](=O)[O-])nc1 CN1CCc2cc(C(N3CC(C4(NC(=O)C=C(Cl)Cl)CC4)C3)=O)sc2C1 N1(C(CNC(C)=O)=O)CCC(C2(Nc3ccc(-c4nnco4)cc3)CC2)CC1 N1(C(C=C(C)c2ccco2)=O)CC2CCCC2C1C(=O)NCC(C)C1CC1 c1(CC)cc(C(F)(F)F)ccc1C(=O)N(CCNC(C1CCCC1O)=O)C1CC1 N1(C(CSc2nc(C)[nH]n2)=O)CC2(CCCC2NC(=O)CC2CCC(O)C2)C1 Cc1ccc(C(N2CC(N(C)C(c3sccc3C(C)C)=O)C(F)C2)=O)c(Cl)c1 C(=O)(CC(C)(C)C)N(CC(C)C)CC(=O)NC(c1nc(C(C)C)cs1)C CC(CC(=O)N(C1CCSC1)C)C(C)(C)NC(=O)CNC(=O)C(C)(C)C S(=O)(=O)(c1cc(C)cnc1N1CCC=C(Cl)C1)NC(CCC=C)CO c1(C2C(C(=O)NCC(CNC(C3CC(OC)C3)=O)C)C2)nc2ccccc2[nH]1 CCC(C)C(C)C(=O)N1CCC(C)(CNC(=O)C=C(C)C(F)F)C1 Cc1cncn1CCC(=O)NCC(C)N(C)C(C1CC1C(c1ccccc1)=O)=O C#CC1(C(=O)NCCC(=O)OC)CCN(C(C2CCN(CC)CC2)=O)C1 C1(NC(C2N(C(C)=O)CSC2)=O)CC(C)CN(C(=O)C(C)Cc2ccccc2)C1 c12c(C)ccnc1N1CC3C(C3C1)NC2=O.c1(C(=O)OC)ccc(F)cc1C CCC(CNC(C1CN(C)C(=O)N1)=O)(CC)NC(c1cc(SC)c(C)o1)=O c1(C(=O)NCC(C(=O)NC(CC2CCCC2)CO)OC)cc(O)nn1C N1(C(C(=O)NCCCOC)C)CCOC(CNC(=O)CCN2CCCC2)C1 C1(CNC(c2c(C)nc(C)o2)=O)CC2CCC(C1)N2C(C1CC1C(C)O)=O C(=O)(C(C(C)(C)C)NC(C1COCCN1C(c1cccc(SC)c1O)=O)=O)NC c1(C(=O)NC2CCCN(C(C(C3CCCC3)OC)=O)C2C)ccn2c1CCCC2 S(=O)(=O)(c1cccs1)NCCC(=O)NC1(CO)CCN(C(=O)C2=CCCS2)CC1 N1(C(c2ccc(C(C)C)o2)=O)CC(F)(F)CC1C.C12CCCCCC1C(=O)N2 S(=O)(=O)(c1ccc(C(N2CCN(C)CC2CNC(C2CC2(C)C)=O)=O)cc1)NC N1(C(C(C(CC)C)O)=O)CC2OCCN(C(c3c(F)cc(F)cc3F)=O)C2C1 Cc1c(C(N2CC3(CC(CNC(c4cc(O)ncn4)=O)C3)C2)=O)cccc1F C1(CNC(C2CCc3nncn3C2)=O)CCCCN(C(C2CCCC2)=O)CC1 N1(C(c2ccc(C)c(C)c2)=O)CCN(C(=O)Cn2cnc(Br)n2)C2CCC12 c1(C(=O)NCCN(CCC)C(C2(C)CCN(C)C2=O)=O)cccc(C)c1F N1(C(CCC=C=C)=O)CCC2(NC(c3ccc(O)c(C(C)(C)C)c3)=O)CC2C1 C(=O)(CC(C)C(F)F)NCCC1(C)CCN(C(Cc2c(C)scc2)=O)C1 c1(NC(=O)Nc2ccc(CC(N)CO)cc2)ncc(C=NO)s1 C(=O)(C(F)(F)CC(C)C)N1CC(N(CC#N)C(c2c(C)cccc2C)=O)C(C)CC1 CCCCC(C(=O)NC1(n2cncn2)CC1)NC(=O)C1=C(Cl)CCC1 CC(O)C(C)(C)C(=O)N1CC2CC(C1)N2C(c1cc(Cl)ccc1C(F)F)=O C(=O)(C(F)(CNC(C1CCC2(CCC2)O1)=O)C(C)C)NC(CC(C)C)(C)C c12cccc(c1)C=CCn1ccnc1-2.Cn1ccc(CCc2ccccc2)n1 c1(C(=O)NCCCN(CCO)C(C2CC23CC3(F)F)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(N(CCC)CCNC(=O)C(C2CCCCC2)O)=O)nccc(N)c1Cl CC(C(C(=O)NC1COC1)N(C)Cc1nnn(C)n1)C1CCCC1 C1(CC)C(C(=O)NCc2ncnn2C)CCN1C(=O)CC1CC(OC)C1 C1(COC)(NC(C23CC(CC(F)F)(C2)C3)=O)CCN(C(C2(C)CNC(=O)C2)=O)C1 C1(CC(=O)NCC(CNC(c2ccc(NC)cc2)=O)OC)CCC(=O)NC1=O Cc1cnc(C(=O)NC2CCN(C(c3ccncc3N3CCCC3)=O)C2)c(F)c1 C1(NC(C(CC2CCCC2)NC(C2N(C)C(=O)CC2)=O)=O)COC2(CCCC2)C1 C1(C(=O)NC2C(O)CCN(C(C3C(OC)CCCC3)=O)C2)CN2CCN1C(C)C2 C(CCN=c1nc(N2CCC(O)CC2)c2c([nH]1)CCC2)c1cccc(C)c1 C1(CC)C(C(N2CCC(C)(CO)C2)=O)CCN1C(C1CCCN1C=O)=O.C(C)(=O)N c1(C(=O)NC(C2CCN(C(=O)C(N3CCCCCC3=O)C)C2)C)cc(Cl)nnc1O N1(C(CC(C)SC)=O)CCN(C)C(CNC(=O)Cn2ccc(C3CC3)n2)C1 N1(C(Cn2c(C)nnn2)=O)CC(CO)C2(C1)CN(C(=O)CC1SC(=N)NC1=O)C2 C(CCC(N)=O)(C(=O)NC1CCCN(C(c2cccc[n+]2[O-])=O)CC1)N(C)C N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C2CN(C(=O)C(COC)OC)C2)C1 C1(CC=C)(NC(C2CC2(C)Br)=O)CCN(C(C23CCC(CC2)C3)=O)C1 CCCC(CNC(=O)C(C)SC)C(=O)Nc1ccc[n+]([O-])c1 Cn1ncc2cc(COC(c3cc([N+](=O)[O-])ccc3CN)=O)ccc12 C(N=c1ccnc(COC)[nH]1)C1C(NC(C(C(C)C)OCCOC)=O)C1(F)F C1(NC(CN(CCCCCC)C)=O)CC2CC(NC(c3ccc(F)cc3)=O)C2C1 c1(OC)cc(C(=O)NCC(C)(O)CNC(=O)CC(C)c2cccnc2)cc(Cl)n1 c1(C(=O)NC2(c3cn(C4C(C)CCCC4)nn3)CCC2)ccc(F)cc1[N+](=O)[O-] c1(NC(CC2C3CN(C(=O)OC(C)(C)C)CC32)=O)ncn2ccccc12 C1(C(N(C)CCNC(=O)CSCCC(F)(F)F)=O)CCc2nn[nH]c2C1 N1(C(CN2CC(C)(C)C2)=O)C2CCC1CC(CCNC(c1sccc1C#N)=O)C2 C#CCCCCCC(=O)NCC1(F)CCN(C(=O)Cn2ncc(Br)c2C)C1 c1(C(=O)NC2(C)CN(C(C=Cc3ncn(C)c3)=O)C2)ccc2c(=O)cc[nH]c2c1 S(=O)(=O)(CC(=O)N(C)CCN(C)C(C1CC2CCCC12)=O)N(CCC)CCC N(C1CN(C(C)=O)Cc2ccccc21)C(C(C1CCC1)OCC)=O N1(C(C2C(OC(C)=O)C2)=O)C2CCC1C(C)C(NC(C1CCC3(CC1)CC3)=O)C2 CCCC(CC)CCC(=O)N(CC(C)(C)NC(c1nccc2occc12)=O)C CCCC(C(C)CC)NC(=O)CC(O)(C(F)(F)F)c1ccccc1 C(=O)(C(CC(F)(F)F)NC(c1cc(F)ccc1OC)=O)NC(CCCCC)C N1(C(C(CC)(CNC(C2CCCCC2O)=O)CC)=O)CCC2(CCOC2)CC1 c1(C(=O)NCC2(OC)CN(C(C(C)N(CC)CC)=O)C2)cncc2ncccc12 Cc1ccc2c(CC(=O)NC(C)CN(C(=O)C#CC3CCCCC3)C)c[nH]c2c1 C(=O)(CC(C)NC(C1(CNC(c2sccc2F)=O)CCC1)=O)OC c1(CN2CC(NC(c3cc(C(C)C)[nH]n3)=O)C(F)(F)C2)ccc2nccnc2c1 C=CCC(C(=O)NCCn1ccc(C(N2CCSCC2CO)=O)c1)C(C)C c1(NC(C(CCCNC(c2cc(OCC)no2)=O)O)=O)cccc(F)c1OC c1(C(=O)NC2CC2CNC(C2CC(F)C2)=O)cncc(-c2ccccc2F)c1 c1(CNC(CC(COC)C)=O)ccc2c(c1)CCN(C(=O)CC(C)OC)C2 c1(C(N2C(CNC(C3CC(O)CN3C)=O)CC(OC)C2)=O)ccn2ccnc2n1 N1(C(c2occ(C(=O)OC)c2)=O)CCC(O)(CCNC(C2(CF)CCC2)=O)CC1 C1(NC(C(OCC)OCC)=O)CCCCC12CCCN(C(C1CC1(C)C)=O)C2 N1(C(C=CC=CC)=O)CCC(C)C(N(C(=O)C=Cc2c[nH]nc2C)C)C1 c1(CN(C(C2CN(c3ccc(Cl)cc3)C(=O)O2)=O)C2CC2)cnc2n(c1=O)CCS2 C1(C(N(CCC(c2cccs2)NC(=O)CC2CCC2)C)=O)CCSC1 c1(C(=O)NC2CCC(CNC(C3(CCOC)CCCC3)=O)C2)n[nH]cc1[N+](=O)[O-] N1(C(C2(CC)CCOC2)=O)CCC2(CCCCN(C(=O)C(=O)NC3CC3)C2)C1 C1(COC)(NC(c2cccs2)=O)CN(C(C2CCC(Cn3ccnc3)O2)=O)C1 c1(C(=O)NCCN(CCC)C(C2CC(C(F)F)(OC)C2)=O)cnc(O)c(Cl)c1 c1(CC)ccc(CSC2(C(=O)Oc3ccc(SC)cc3)CNC2)c(F)c1 N=c1nc2c(c[nH]1)CN(c1nc3c(s1)CC(c1ccccc1)CC3)C2 c1(C(=O)NCC2CCCCO2)cccc(CSCC(CO)NC(C2(Cl)CC2)=O)c1 N1(C(CC(=O)NCC)=O)CCCC(N(CCSC)C(C2CCOCC2)=O)C1 C1(C(N2CCC(NC(c3n(C)ncc3Cl)=O)C2)=O)CC2(CCO1)CC2 c1(C(=O)NCC(C(=O)NC2CCN(C)C2=O)N(C)C)cc(N)cc(F)c1 CC1=NOC(C(N2CC3CC2(CNC(=O)CCN2C(=O)CCC2=O)C3)=O)C1C C1(CNC(C(CC)F)=O)CCC(F)(CNC(=O)CCC2CC2C)CC1 C1(CC(=O)OC)CC2C=CC1C2.n12cc(cn1)C(CC(N)=O)NCC2 Nc1ccc(C(=O)NC2CCCCC2NC(=O)C(F)CC2CCCC2)c(F)c1 C(C(C)(C)C1=CCOCC1)NC(c1ncc(Br)cc1F)c1n(C(CC)C)nnn1 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(C)N(C(c2n[nH]c(C)c2O)=O)CC1 C=CCN=C(NCC(N1CCCCC1)=O)N1CCC(C)C1.N1(CC)CCC(C)CC1 CC(C)CC(C(=O)NC(Cn1cccn1)C(N1CCC(C(C)C)CC1)=O)C(C)C CCC(O)C(F)(F)C(=O)N1CC(CNCc2cn(CC(=O)OC)nn2)C1 c1(C(C(N2CCC(CN(C(=O)Cc3ccco3)C)C2)=O)(C)C)cccc(Cl)c1F N1(C(CNC(C(C)(C)C)=O)=O)CC2(CC(CC(=O)NC(=N)O)C2)C1 c1(N(CC(C)(F)F)C)ccncc1S(=O)(=O)NC1CC(C)(C)CC(C)(C)C1 c1(C(=O)NCC2(NC(c3n(C)cnn3)=O)CC2)ccc(-n2ccnc2)nc1 N1(C(c2nc(C)sc2C)C(=O)NC(CC)C)CCC2(CC1)CC(O)C2 c1(C(=O)Nc2cccc(NC(c3n(C)ncc3)=O)c2)cnc(Cl)cc1Cl C(CCC(C)CN1CCCC(C(=O)O)C1)=C(C)C C1(CNC(c2c(C)ocn2)=O)CCC2(CC1)CCN(C(=O)C=C1CCC1)CC2 C1(NC(C(CCOC)C)=O)C(C)(C)C(NC(=O)CSS(C)(=O)=O)C1(C)C C1(CC(C)CO)CCN(C(C(=O)NCCC2(C)CC2)c2cccs2)CC1 C(=O)(C(C)S(C)(=O)=O)NC1CCN(C(c2c(C)cco2)=O)C1c1ccccc1 C1(NC(C2CC(C)C2)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC1(C)C c1(OC)ccc(C(N2CCC(NC(C3CC=CC3)=O)C(C)C2)=O)cc1[N+](=O)[O-] N1(C(c2ccc(CC)cc2N)=O)CC(C2CN(C(=O)C(c3ccccc3)F)C2)C1 N1(C(c2ccn(CC)n2)=O)CC(C(N2CCC(C3CC3)CC2)=O)CC(C)(C)C1 CCS(=O)(=O)CC(=O)NCCC(N1CC(O)C(F)C1)=O Cc1cc(C)c(C(=O)NC2CC(C(C)NC(C3CCCN3C=O)=O)C2)o1 c1(C(=O)NC2CN(C(CC=CC)=O)CC(O)C2)cccc2c1CCCC2 c1(CCOC)nc(C)cc(=NCC2COCC(C)(C)C2)[nH]1 c1(NC(N(CCCCO)C(C)C)=O)ccnn1CCN(C)C C(CN=c1[nH]nc(C(F)F)s1)N(c1cccc(OCC)c1)CC C1(C(C)C)C(NC(c2cnn[nH]2)=O)CCN1C(c1ccc(NS(C)(=O)=O)nc1)=O C(C(C)(O)CC(=O)NC1(C(=O)NC2CC3CCCC3C2)CC(O)C1)OC c1(CN2CC(C(=O)NCC=Cc3ccccc3)SCC2)cc(Cl)ccc1Br C1(C(=O)NCC(CNC(CNC(CCCCC)=O)=O)(C)F)CCC2(C1)CC2(F)F C#CC1(C(=O)NCC(C)(CO)NC(=O)COc2c(C)occc2=O)CCOCC1 c1(OC)cc(OC)c(OC)cc1-c1nccn1C1CCNC1.N1(C)C(=O)CCC1=O N1(C(C=C(C)CNC(C2CC(CF)C2)=O)=O)C2CCC1CN(C)CC2 c1(C(=O)NCCC(C)N(C(c2c(OC)ccs2)=O)C)cnc2n1CC(C)CC2 Cc1nc(-c2ccccc2F)sc1C(N1CC(CC(C)NC(C2(C)CC2)=O)C1)=O C=CCC(CC)C(=O)NCC(C)(C)CC(=O)N1CCC(n2cncn2)C1 C1(C(=O)NCC(C)NC(C(C)Sc2ncccn2)=O)CC(=O)C1(C)C N1(C(CN(C)CC)=O)CCN(C(c2nncs2)=O)C(c2ccc(OCCO)cc2)C1 C1(C(=O)NCC2CN(C(C)C)C2)CCN(C(C2CCCC23CCC3)=O)CCO1 C#Cc1ccc(C(N2CC(N3CCN(C(=O)C(C)n4ccnn4)CC3)C2)=O)cc1 C(=O)(C(C)CC(=O)N1CCCC(CNC(=O)CNc2cnccc2C)CC1)OC N1(C(Cc2cc(C)sc2C)=O)CCCN(C(=O)COc2ccsn2)CC1CO N1(C(C(C)OC2CCOC2)=O)CC(NC(=O)Cc2ccnn2C)C(C)(C)C1 N1(C(C2CC(c3ccccc3)(NC(CC3CN(C)C3)=O)C2)=O)CC2CC1C1CC21 Cc1cccn2c(Br)c(CN3CCCC3c3cccc4c[nH]nc34)nc12 c1(CC(=O)N(CC(C)O)CCNC(c2c(C#C)c[nH]n2)=O)cc(C)cc(F)c1 N1(C(CC(CCC)C)=O)CCCN(C(c2cnn(CC(F)(F)F)n2)=O)C(CO)C1 CCC(C#N)(CC)C(=O)N1CCCC(C)(NC(c2nnc(C)s2)=O)C1 C(=O)(CCC(=O)NC(C)C(C)NC(c1ccn(C2CCCC2)n1)=O)NCCC N1(C(C)=O)CCCC(CN2CC(OCCO)C2)C1c1cnn(C)c1 c1(C(N(CC(=O)NCC2(O)CCC(C)C2)C2CCC2)=O)ccn2ccnc2c1 c1(CC(=O)N(C)Cc2ccccc2)cccc(=O)n1C.C1(=O)C(N)CN1 C(=O)(C(O)CC(F)(F)F)N(CCN(C(c1cncc(C2CC2)c1)=O)CC)CC C1(C(N2C(C#C)CC2)=O)CC2CCC(C1)N2C(c1cncc(C#N)c1)=O C(=O)(CCC(C)(F)F)N1CCCC(CNC(COCCN(C)C)=O)C1 C1(C(=O)NC(CN(C(C)C)C)C)CCCN(C(C2CC3(CSC3)C2)=O)C1 c1(C(N=c2nc(C)[nH]s2)=O)cnc2c(-c3ccc(N(C)C)cc3)cnn2c1 N1(C(CCc2n[nH]c(C)c2C)=O)C2CCC1CN(C(c1n[nH]cc1[N+](=O)[O-])=O)C2 CC1=CCC(NC(c2cc(CC3CCN(C(CCC(C)C)=O)CC3)oc2C)=O)CC1 C1(C)(CCC(=O)NCC(C)(CO)NC(C2C(c3c(C)occ3)C2)=O)CCC(=O)N1 CC1CC(NC(c2cc(Cl)ccc2F)=O)CN(C(=O)CN(C2CCSC2)C)C1 c1(NC)cnncc1C(N1CCC(CCC(=O)NC(C2CCCO2)CO)CC1)=O Cn1ccc(C(=O)NCCN2CCC(NC(=O)C(=O)NCCC(N)=O)CC2)cc1=O C1(CNC(CNS(CC)(=O)=O)=O)CN(C(=O)Cc2c(C)n[nH]c2C)CC12CCC2 c1(C(C)C(=O)NCC(C)NC(=O)C(c2cccc(N)c2)O)cccc(F)c1 C(=O)(C#CC(C)(C)C)NC1CN(C(c2c(CC)cccc2)=O)C(COC)C1 c1(C(c2nnnn2CC)NCC2CCOCC2)cc(CC)ns1 C1(CCC)CC(C(=O)NCCN(C(=O)Cc2ccccc2SC)C)CCO1 C(=O)(C(CC(C)C)n1ccnc1)N1CCCC(N(C(CC)=O)CC2CSC2)C1 CC(C)C(F)C(=O)NC1CCC(NC(=O)CCOc2cccnc2)C1 C1(N(C)C(C2C(c3ccccc3)C2(C)C)=O)CCN(C(C2(C)CC=CCC2)=O)CC1 N1(C(c2cnc(CC(C)C)s2)=O)C(C)C2CC1C2NC(c1cccs1)=O C1(CNC(C(CC)COC)=O)CN(C(=O)CN2CCCCCC2)CC1(F)F Cc1cc(C)n(CC(=O)NC2CCC2NC(c2cnn(CCF)c2)=O)n1 N1(C(C(C#C)(C)C)=O)CCCC2(NC(C3CCC(=O)N(C)C3)=O)CC2C1 C1(C(=O)NCC(CC)NC(=O)CC2(C)CCCO2)CC(C2CCCC2)C1 N1(C(CCC)=O)CCc2c(NC(=O)NNC(=O)c3ccc(=N)[nH]c3)cccc21 c1(CN2CC(C(N(CC(C)C)CC(C)C)=O)C(C)C2)cccc(=O)n1O C1(NC(C=CCOC)=O)CCCOC12CCN(C(=O)C#CC(C)C)CC2 C1(CN)C(C(=O)O)CCN1C(c1cn(-c2ccccc2)nc1C(C)C)=O c1(-c2ccc(CN(C)CC3CC3)s2)cc(C2CC2)ccc1F.CC1CCC(=O)N1.CCO c1(CNC(=O)NC(c2ccc(C(C)C3CC3)cc2)C)cc(Br)nn1C c1(C(=O)NC2CCC(C)N(Cc3ccc(F)c(F)c3)C2)nc[nH]c2ncnc1-2 CC1CCC(CNCCCOc2ccncc2)CN1 Cc1cnc(Cl)c(C(N2CCOCC(CNC(=O)Cc3sc(C)nc3C)C2)=O)c1 c1(CC)cc(C(N2CCC(C(=O)N(C)CC3COCCO3)C2)=O)ncn1 N1(C(C(CC#C)C)=O)CCC2C1CCCN2C(=O)CN(CC)CC C1(NC(COCCCCC)=O)CN(C(=O)C(C#N)(CC)CC)CCC1(C)C C1(=C(C(=O)N(CC(=O)N(C)CC2CCC2)CC#C)C)CCC(C)CC1 c1(C(=O)NCC2(CNC(=O)CO)CC2(F)F)cccc2cccnc12 CCC(C)(C)C(O)C(=O)NCC1C2CN(C(C34CCC(CC3)CC4)=O)CC12 C12(NC(CC(CC=C)NC(=O)CN3CCCC34CCC4)=O)CCC(O)(CC1)CC2 CC1CCc2[nH]nc(C(=O)NC3C4CC3N(C(c3cc(C(N)=O)c[nH]3)=O)C4)c2C1 C1(C(=O)NC(C)CCCCNC(c2cnco2)=O)Cc2cncn2C(=O)N1 N1(C(C(COC)NC(c2ccnc(O)c2F)=O)=O)CCCC2CN(C)CC12 C12(C(=O)NCC(C3CC3)NC(c3ccnn3C3CCC3)=O)CCCN1CCC2 CC1(C)CC(C)(CO)CN1C(C1CCCCN1C(c1ccc2n[nH]cc2c1)=O)=O C1(C(=O)NCC(CNC(c2cccc(N(C)C)n2)=O)(C)O)CC2CCC1CC2 c1(C(=O)NCCC2N(C(c3c(C)cn(C)c3)=O)CCSC2)c(C)ncn(C)c1=O C(=O)(C(CCC(C)SC1CCOC1)N1CCC(CO)CC1C)NC1(CSC)CC1 C1(N(C)C)CCCC(NCc2ccccc2OCC#N)C1 N1(C(=O)NC(COC)C)CCC2(CC1)COC(C)C2N C(CNC(c1cnn(CC)c1Br)=O)(CC(C)C)NC(C1C(=C)C1)=O c1(CC(=O)NC2CC(CC)C2)nnc(C)s1 c12nc3c(s1)CC(CC3)NC(=O)c1n(nc(C3CC3)c1)C(C)N2.C1(NC)CC(O)C1 C(=O)(C(F)CCC(C)(C)C)N1CCC(C(C(=O)Nc2c(OC)nsc2)C)C1 c1(C(=O)NCC(C(C)C)(C)NC(=O)CSc2nnnn2C)nc2c(s1)COCC2 C1(CCCNC(c2ccn(C)c2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCO1 c1(C(N2CCCC23CCN(C(=O)C(F)CC2CC2)C3)=O)cc2ccc(Br)cc2cn1 N1(CCC=C)CCC(C2CC(NC(=O)CO)CCO2)CC1.N12CCCCC1C2=O C(C(O)C(=O)NCc1conc1C(C)C)NC(C=C(C)C(C)C)=O N1(C(C=CC)=O)CCC2CN(C)CCC12.c12cnc(nc1)C(=O)NC1(CCC1)C2 C1(NC(Cc2c(C)noc2)=O)C=CCN(C(=O)C(C2CCCCC2)F)C1 C(=O)(C1=CS(=O)CCC1)NCCN(C(c1c(C)noc1C)=O)C CC1C(NC(C2CCCOC2c2ncc[nH]2)=O)CCCN1Cc1cnn(C)c1 N1(C(c2c(F)ccc(C#C)c2)C(=O)NC(C)CC)CC2(C)CN(C)CC2(C)C1 C1(C(=O)NC(CC)(C)CO)CC=CCC1NC(=O)CC1CC2CC2C1 c1(C(=O)NCCC)ccc(CS)o1.C(c1cnc[nH]1)=C(C(=O)N(C(C)=O)CC)C N1(C(C(C2CCCC2)NC(CC(=O)OCC)=O)=O)CCC(C)=C(C)C1 N1(C(C(C)NC(CC)=O)=O)CCCC2(NC(c3cc(CC)nn3C)=O)CC2C1 C1(CN(C(C(C)CO)=O)C2COC2)CCN(C(=O)CCF)CCC1(F)F c1(NC)nc(C)ccc1C(N1CC(CC(C)NC(C2CC(=O)N(O)C2)=O)C1)=O C1(C(=O)NC2CCC(n3cc(C(C(C)C)(C)C)nn3)C2)C2CC3C(C2=O)C13 N1(C(C2(C(F)F)CC(=O)C2)=O)CCC2CN(C(=O)C(F)C(F)(F)F)CC2CC1 c1(C(N2CCCC(C(C)NC(c3c[nH]ccc3=N)=O)C2)=O)ccc2c[nH]nc2c1 CCCCS(=O)(=O)NC(C)C(=O)NC1COCCC1NC(=O)CC(C)C c1(C(=O)NCC2CC(C(F)(F)F)C2)cccc(Oc2ccc(Cl)cc2)c1 C1(NC(c2cc(CC)on2)=O)CCCCC12CN(C(C1CNC(=O)O1)=O)CCO2 c1(NC(c2ncc(C(F)F)s2)=O)ccc2c(c1)CCN(Cc1ccc(O)nc1)C2 CON(CCC(=O)N1CCC(C)(O)CC1)C(=O)CCc1cn(C)cn1 C=CCC(C)C(=O)NC(C)CC1CCN(C(C2OCCOC2C)=O)CC1 c1(CNC(COC)=O)cnn2c1CN(C(c1c(C)cc(O)cc1C)=O)CC2 C1(C(N(CCN(C(C)C)C(c2coc(C(F)F)c2)=O)C)=O)CCC(O)C1 c1(C(=O)NCC(C)(C)NC(=O)C2CC2)nnn(-c2ccc(F)cc2)c1C(F)F C(=O)(CCC(=O)NCCC(C)CCNC(=O)CSCc1nc(C)no1)OCC n1(CCN2CC(O)CC2)cc(C(=O)N(C)C)cn1.CCOC N1(C(C(C)=C(CC)C)=O)CC(CNC(c2cc(COC)cn2C)=O)C(C)(C)C1 c1(C(=O)NCCNC(C2CCCC(OC)CC2)=O)cnn2cc[nH]c(=O)c12 N1(C(C2(COC)CCCO2)=O)CC2(CCCCN2C(C2CCCCC2O)=O)C1 C1(CC)CCCN(C(c2cn(C)nc2OC)=O)C1C(N1CCSCC1)=O N1(C(C(CC)C)=O)C2CCC1C(CNC(c1csc(-c3ccoc3)n1)=O)C2 c1(OC)ccc2[nH]cc(C(=O)NC3CC3NC(=O)CCc3cnccn3)c2c1 C1(NC(c2ccc(CSC)o2)=O)CC2CC(C1)N(CCNC(C1CC1(C)C)=O)C2 N1(C(C(C)C2CC2)=O)CC(NC(=O)Cc2ccn(-c3ccccc3)n2)C2(CC2)C1 C1(C(C)NC(C2(F)CC2(Cl)Cl)=O)CN(C(=O)CC(c2cccc(F)c2)O)CCO1 CN1CCCC1CC(=O)NC1CCC(CCNC(=O)CNC(c2ccsc2)=O)C1 c1(CC(N2CC(O)(CNC(CCC=C)=O)C2)=O)ccc(C#N)cc1 CCC(CNC(=O)C(=O)NCCc1ccnc(C)n1)(CC)CCO N1(C(c2cnc(C(C)O)s2)=O)CCCC2(NC(=O)C=CI)CC2C1 c1(OC)ncc(Cl)cc1C(=O)NCC1(C)CCCN(Cc2cc(C)nc(O)c2)C1 N1(C(CCSc2n(C)ccn2)=O)CCC2(NC(C3(C(=O)N(C)C)CC3)=O)CC2C1 N1(C(=O)NC2C(C)COCC2)CCC2(CCCCN2C(=O)OC(C)(C)C)C1 C(CCCCCC(=O)NCCN1CCCC1=O)NC(C(C)(C)CCF)=O C1(CCNC(C2C(CNC(C(CSC)OC)=O)C2)=O)CCC(C)(C)C1 N1(C(C(c2cccnc2)C)=O)CCC(CNC(C2CCC(=O)N2)=O)C1 C(C(C)(C)C(=O)OC)N(CCCOCC(=O)NCC)CC1(SCC)CC1(F)F Cc1ccc(C(C)NC(=O)CCNC(c2cnco2)=O)cn1 C1(C2CCN(C(c3c(-c4cccs4)nc(C)s3)=O)CC2)CC2CCC1CC2 N(C1CN(C(=O)CS(N)(=O)=O)Cc2ccccc21)C(c1c(OC)ncc(F)c1)=O c1(C(=O)NCC(C)(C)CNC(c2csc3cncn23)=O)c(N)cccc1Cl c1(C(=O)NCCC(C)NC(C2(C#N)CCCO2)=O)c[nH]c2cccc([N+](=O)[O-])c12 Nc1cc(C(N2CC3(C2)CN(C(=O)CC2CCSC2)C3)=O)ccc1F c1(-n2cc(C3(C(c4csnn4)=O)CCC(C(F)F)C3)nn2)cccc([N+](=O)[O-])c1 CC1C(C)N(C(c2ccsc2-n2cnnn2)=O)CCN1C(C1(O)CCOCC1)=O c1(CC(=O)N(C(C(C(C)C)OC)c2ccccc2)C(C)C)cc2ccccc2s1 c1(SC)ccc(Cl)c(C(=O)NCCC2(O)CCN(C(c3cccnc3)=O)CC2)c1 N1(C(C2CCC3(CCC3)O2)=O)Cc2n[nH]cc2C1C(=O)N1CC(F)C(F)C1 c1(C(=O)NC(C)CNC(=O)CSC2CCCCO2)cc(O)nc(O)c1 N1(C(C(C)N(C(C)=O)C)=O)CC2CC(N3Cc4c[nH]nc4C3)C1C2 c1(C(c2nnnn2CC(F)F)NC2C(C)C2C)ccc(Br)c(Cl)c1F Cc1cc(C#N)ccc1C(=O)N(CC(=O)N(C12CC(C1)C2)C)CCO C1(C(=O)NC(CCOC)CNC(c2cscn2)=O)CCCN(S(=O)(=O)CCC)C1 c1(CC(=O)NCC2(OC)CN(C(=O)Cc3ccccc3Cl)C2)ccc(F)c(Cl)c1 C(=O)(C(CC(N)=O)NC(=O)CC(F)(F)F)NC(C(=O)NCC)C C(=O)(C(C#N)C(=O)C=CC1CCCO1)N(CC(C)C)C(C)C c1(C(=O)NCC2N(C(c3occ(C)c3C)=O)CCCC2C)ccc2nccn2c1 C1(CC(=O)NC(C)CCCO)CCN(C(=O)C(=O)N(C)C)CC1 Cc1cnc(C(N2CCC(O)(C(C)NC(=O)CC3COCCOC3)C2)=O)cc1C c1(NC(C(C2(O)CCCCC2)NC(C2COCCO2)=O)=O)cccn2nccc12 C1(NC(C(C)C(F)F)=O)CC2CCC1CN2C(=O)Cc1cnns1 C12CCCN(CC1)C(=O)CCn1cc2nn1.c1(CC(=O)OCC)ccnc(F)c1 C1(NC(c2ccc(NC=O)cc2)=O)CC2CC1N(C(c1cc(Cl)ccn1)=O)C2 c1(C(=O)NC(C2CCOC2)CNC(C(CC)CC)=O)cc(C)nc(C(F)F)n1 c1(C(=O)NC(CN(C(c2c(C)cncc2C)=O)C)C)cccc2oc(=N)[nH]c12 C#Cc1ccc(C(N2CCCC(CCNC(=O)CC3CCCC(C)O3)C2)=O)cn1 C1(NC(CC2CC(NC(c3c(C)nns3)=O)C2)=O)CC2(COCCO2)C1 C(=O)(C1=C(Cl)CCC(C)C1)N1C(C2(O)CN(C(c3nc(CC)oc3C)=O)C2)CCC1 N1(C(c2c(C)c(N)n(C)n2)=O)CCOCC12COCCN(C(=O)C=C(Cl)Cl)C2 C1(CC)CC(C2C(=O)NCCCC3(CCC3)N2C)C1.c1(C(=O)OC)ccco1 N1(C(CC2(CS(C)(=O)=O)CC2)=O)CC2(NC(C3CCCO3)=O)CC1C2 N1(C(C(Cn2cccn2)NC(=O)CC2C3CC4C(C3)C24)=O)CC2CCCC12 C1(CNC(=O)CCN2CCC(F)C2)CCCC1NC(c1ccn(C2CCC2)n1)=O CC1CN2CCCC2CN1C(=O)C#CC(C)(C)CNC(=O)CC1CCCC1 c1(NC(C)=O)ccc(C(=O)NC2CCC(N(C(=O)C=CC3CC3)C)C2)cc1F C1(CNC(c2c(C)nco2)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1(F)F CN1CCN(C(C2CS(=O)(=O)CC2N2CCCC2)=O)CC1c1nn[nH]n1 C1(NC(C(C)OCCOC)=O)Cc2ccccc2C1NC(C1CCCCC1C)=O C(=O)(C(F)(CNC(=O)C(C)C(=O)OC)C(C)C)N1CC(C#C)C(OC)C1 C(=O)(CC(C1CC1)NC(c1cc(Cl)no1)=O)NC(CC=CC)C C(=O)(CC(C(F)F)C(C)(C)C)N1CCC(N(C(=O)C=C2CCC(C)C2)CC)C1 CC1CCCN1CC(=O)NC(C)CCN(C(=O)CSCc1ccccc1)C C1(NC(=O)CCN2CCC2)CCN(C(C2(c3cc(Br)ccn3)CC2)=O)CC1 c1(C(N2CCN(C(C)=O)C(C)C2)=O)cc(C)c(C)[nH]c1=O Cc1nn(-c2ccc(F)cc2)c(C)c1C(=O)NC(CNC(=O)C1=CCOC1)CO C1(C(N2C(CNC(CC(=O)OCC)=O)CC2)=O)CC(C)CCC1C(C)C c1(CC(N2CCCC(NC(c3scc(C(C)=O)c3)=O)C2)=O)cc(C)ccc1F CCCC(O)(Cn1ccnc1-c1ccc(SCC)c(Cl)c1)CCC c1(OC)cnc(C(N2CCC(NC(=O)C3=CCOC3)C(O)C2)=O)c(F)c1 N1(C(CCCC(C)NC(C(CC)(C)C)=O)=O)CCCCCCCC1 C1(C(=O)NC2CC(C(C)NC(=O)CC3CC4CC4C3)C2)CCC(C)(C)O1 C1(NC(C2CC3(CCCC3)CO2)=O)CN(C(C2C=CCC2)=O)C2CCCCC12 C1(C(N(CC(C)CNC(=O)Cc2cccnc2)C)=O)CCCCNC1=O C12(C(C)N(C(CC3N(C(c4c(C)csn4)=O)CC3)=O)C3CC3)CCC(CC1)C2 c1(OC)cc(Cl)ccc1C(=O)NC1(CF)CCN(C(=O)C(F)OC(F)(F)F)C1 N1(C(c2cc(C)oc2)=O)CCC(C)(C)C1CNC(C12CCCC1C2(F)F)=O C1(C(=O)NC2CC(=C)C2)CN(C(c2nc(COC)oc2C)=O)CC1(C)C C1(O)(CN(C(C2(CC#C)CCOC2)=O)C)CCN(C(=O)CCC2CCOC2)CC1 O(NC(=O)CCCCCNC)CCNC=O.C(=O)(C(C)CC=CC)CC#C N1(C(c2ccn(C(C)C)n2)=O)CCC(O)(CNC(C2OCC2(C)C)=O)C1 C1(C(C)C)CN(C(C2COCC2C(F)F)=O)CCN1C(c1nncn1C(C)C)=O c1(C(=O)NC2CCCC(NC(c3cc(CCOC)on3)=O)C2)cc2n(n1)CCO2 C#Cc1cc(C(=O)NC2CN(C(=O)CC3(CC)CCC3)CC2SC)cc(F)c1 c1(SC)cc(C)c(C(=O)NCC(C2CC2)N(C(=O)CC2NC(=O)NC2=O)C)o1 c1(C(N2CC(O)CC2C2CC2)C(=O)NC)ccc(-c2cc[nH]n2)cc1.O c1(C(C(=O)NCCCC)N(c2sccc2OC)C)ccc([N+](=O)[O-])cc1Br C1(NC(C(C)n2ccnc2)=O)CC2(C1)CC(NCc1ccnnc1)C2 c1(C(N(C2CCN(C(CCC=C)=O)C2)CC2CC2)=O)cnc2sc(C)c(C)n12 CCCN=C(NCC1COC1)NCC(c1ccc(F)cc1F)CC(F)(F)F C(CCC(O)C(=O)NCc1cnc[nH]1)NC(C=CC(C)(C)C)=O C1(C(=O)NC2(CC=C)CN(C(C3(CC)COC3)=O)C2)CCCCC12CC2 N1(C(CC2C(C(=O)OC)CC2)=O)CC(NC(c2ccc(C(C)C)o2)=O)C(C)C1 c1(C(N2CCC(C)(CC(=O)Nc3ncco3)CC2)=O)cc(Br)cc([N+](=O)[O-])c1Cl CC1(C(=O)NCC(CC2CC2)CO)CC(O)CN1C(c1ccsn1)=O N1(C(C(C)OCC=C)=O)CC(C(=O)N(CC(C)CC)C)C(CCC)C1 C1(C)(C(=O)NCC(C2CCC2)OCC)CCN(C(c2ccco2)=O)C1 C=CC(CCC)CC(=O)NC(C)(C)CNC(C=C(CC)C)=O.OC Cc1ccc(C(N2CC(N(C)Cc3csc([N+](=O)[O-])c3)C2)=O)c(C)c1Br Cc1ccc(CN(C(=O)C(CNC(=O)C(C)OCC(C)C)N(C)C)C)nc1 c1(C(=O)NC(CC)CNC(=O)C(O)Cc2[nH]cnc2C)ccc2nnc(O)n2c1 CCCC(CCC)CC(=O)N1CCC(CN(C(=O)CNS(=O)(=O)NC)CC)C1 C1(C(C)NC(C=COCC)=O)CCN(C(c2ccc(CC3CCCC3)[nH]2)=O)CC1 CN=S(C)(=O)c1cccc(C(=O)NCCCCC(C)NC(=O)C(C2CC2)OC)c1 Cn1nc2c(c1NC(C1CC1C(=O)Nc1cc(F)cc(I)c1)=O)CCC2 Cc1nc(CC(=O)NCCN(CC(C)O)C(=O)CC2(C)CC2(Cl)Cl)c(C)s1 c1(C(=O)NCC(CNC(C2(C)C(C)(C)C2)=O)O)cc(N)c(F)c(F)c1Br c1(OC)cccc(C(=O)NC2CC(O)(CNC(c3ccc(F)cn3)=O)C2)n1 c1(CN2CC(C)SCC2)c(I)ccnc1F c1(CC(=O)NCC(CNC(COCC)=O)F)cc(Cl)n(C)n1 N1(C(c2cc(C)c(C)nn2)C(=O)NC2CC2)CCc2cccc(C)c21 N1(C(Cn2cc(CCCC(C)O)nn2)=O)C2CCC1CCC2.C(=O)(C(C)C(C)O)OC c1(C(=O)Nc2ncc(-c3ccc(CC)s3)s2)c(Cl)c(C)nn1C C1(C(N(CC#C)C)=O)CCN(C(=O)CC2COCCO2)C12CC2 C1(NC(CC2C(C)=NNC2=O)=O)CCCCCC1C(=O)NC(C)C(=O)N(C)C c1(C(N2CC(C)N(c3cc(N(C)C)ncn3)CC2)=O)ccc2ccoc2c1 C1(COC)CCCN1C(=O)C(C1(C)CN(C(=O)C(c2ccn(C)c2)C)C1)C CC1CN(C(C2CNC(=O)N2)=O)CC(C)N(C(=O)CN2CC(=O)NC2=O)C1 CC(C)CC(CNC=O)CC(=O)NC1CCCN(C(=O)CC2(O)CCCOC2)C1 C#CCC(CC(=O)NCCn1cnnc1C)NC(=O)CCCC1CCCO1 C(=O)(CCC(=O)c1cccc(N)c1)NC(C)CCNC(c1c[nH]nc1Br)=O C1(C(=O)NC2CCC3(C(C)C)C2C3)CCN(C(C2(CCF)CCC2)=O)CCO1 N1(C(C2N(Cc3cc(NC(C)=O)cc(OC)c3)CC2)=O)CCC2(CCC(OC)C2)C1 C1(C(=O)NCCCN(C(C(CC=CC)CC)=O)C2CC2)CCn2cncc2C1 C(=O)(CCCCCSC)NCC(CC)NC(=O)CC(C)c1ccncc1 c1(C(C)C)cnc(O)c(-c2nc(-c3ccncc3)nn2CCF)c1 c1(C(C(=O)Nc2ccccc2)N(CC(CCC)C)C)sc(C(F)(F)F)nc1C N#Cc1cccc(C(N2CC(F)(F)CC2CNC(=O)C(=O)NCC(F)F)=O)c1 Cc1ncc(C(=O)NC2C3CN(C(=O)CC4CS(=O)(=O)C4)CC23)cc1C(F)(F)F c1(OC)cc(OC)c(C(=O)NCC(C)(O)CNC(=O)CC(O)CC2CC2)cn1 c1(C(=O)NCCN(C2CC2)Cc2cc(C#N)ncc2)nc2ccccn2c1F c1(CC(=O)NCc2ccncc2)ccc(-c2cnn(C3CC3)c2)cc1.C(=O)N CC1C(C(N2CCCC2CN(C)C(c2ccc(CC=CCO)cc2)=O)=O)CCN1C Cc1ncccc1C(=O)NCC1CC(CNC(C2(C(C)(F)F)CC2)=O)CO1 n1(CC)ccc(=NC(=O)CC2CC(=O)N(C(C)(C)C)C2)[nH]1 Cc1cc(C(N2CC(NC(=O)CC3CC4(CC4)CO3)CC(C)C2)=O)cc(N)c1 N1(C(c2cc(CCC)oc2C)=O)CC2(CCCC2NC(c2ccc(F)cc2)=O)C1 c1(C(=O)NCC(C)CN(C(=O)C(O)c2ccsc2)C)n[nH]cc1Cl N1(C(CCNC(=O)CO)=O)CC2(CCC2)CC1C(=O)NC1CCn2cnnc2C1 C=CCC(CC)C(=O)NC1CC(C)(C(=O)NC2CCCC(C)(C)C2)C1 N1(C(COC(N)=O)=O)CC2(C1)CN(C(C1(c3ccccc3)CCCO1)=O)CCO2 N1(C(C2C(CC)C2)=O)CCC2CCC(C1)N2c1ccnc(C2CCCC2)n1 N1(C(C=CC(=O)NCc2ccc(F)o2)=O)CCN(C(c2cccs2)=O)CC1 c1(C(N2CCC(NC(CCCC=C)=O)C(CC)C2)=O)ccc2snnc2c1 C(C(C)(C)C(=O)N1CCCC(C(C)NC(=O)CCc2ccn(C)n2)C1)N(C)C C1(NC(=O)C(C)NC(C2C3(CC(NC(=O)C4CC4)C3)C2)=O)COC2(CCCC2)C1 CC(=O)CCCC(=O)N1CC2CCC2(NC(c2ccn3ccsc23)=O)C1 N1(C(C(C)Cn2ccnc2)=O)CCN(C(=O)Cc2cn[nH]c2)C(C2CCC2)C1 c1(NC(=O)NC2CCN(C(CCCC#CC)=O)C2)ccc2nc(O)cc(O)c2c1 c1(C(=O)OC)cc(C(N2CC(NC(C3CCC(C(N)=O)O3)=O)C(O)C2)=O)c(C)s1 C1(C(=O)N(C)CCSC)(COC)CCCN1C(=O)C(C(C)C)OC1CCC1 c1(C(=O)NCC2(F)CCC(CNC(CC(C)F)=O)C2)n[nH]c2c1CCSC2 C=C=CC(C)C(=O)N1CC(CCO)(NC(c2cnn(C(C)C)c2Cl)=O)C1 C1(NC(C=CC(CC)=CC)=O)CC2(C1)CC(CNC(=O)CC1COCC(C)(C)O1)C2 C=CCC(F)(F)C(=O)N(C)CCN(C(=O)CC(C)n1cnnn1)C N1(C(C(C)(O)C2CC2)=O)CCCC12CCN(C(C1(C(F)F)CC(F)(F)C1)=O)C2 C1(NC(c2cnc(C)nc2)=O)CC2(C1)CN(C(=O)CN(C)S(=O)(=O)N(C)C)C2 C12(CN3CCC(OC)C3)CCCN1CC(Oc1nccc(N(C)CC)n1)C2 c1(C(N2CCC(COC)CC2)=O)ccnc(N(C(=O)C(C)C2CC2)C)c1 C1(C(=O)NC2CCCC(NC(=O)CC=C(C)C)C2)(COC)CCC(=O)N1 c1(NC)cc(C(N2CCC(F)C(NC(c3ocnc3C)=O)C2)=O)cc(Cl)n1 c1(OC)c(C(N2CC(N3CCCCC3)C2)=O)cnn1C.c12cccc(n1)NC2 C1(CC(=O)NCCCCCCNC(C2CCCC(=O)N2)=O)CCCC2(CCC2)O1 c1(C(=O)NCCCNCc2cc(C#N)ncc2)cccc2oc(O)nc12 N1(C(C(C)N2CCCC2)=O)CC2CC1CN(C(C1CCCCCCN1)=O)C2 C(=O)(C1CCc2cccnc21)NCC(C)(CNC(=O)CCS(N)(=O)=O)OC c1(CC(=O)N(C)CC2CCOC2)ccc(Br)cc1Br c1(C(N2C(CN(C(=O)Cc3ccccc3Cl)C)CC(F)C2)=O)csc2nccn12 Cc1csc(C(C)C(=O)NC2CC(NC(=O)Cn3cc(C4CCOC4)cn3)C2)n1 C(C1CCN(C(C2CC23CCCCC3)=O)CC1)=CC(=O)NC1(C(C)C)CCOC1 CCCC(C(O)C(=O)NOCC(F)F)NC(C1CCC(=O)C1)=O N1(C(CN2CC(C)C2)=O)CCC(CCCCNC(c2cc(F)n[nH]2)=O)CC1 C=C(C)CCCC(=O)NC(C)CC1CCN(C(c2c(Br)cnn2C)=O)CC1 CC(C(C)(C)O)NC(=O)C(C1CCCO1)NC(=O)CCOC1CCCC1 CS(C)(=O)=NS(=O)(=O)NC(=O)COc1ccc(Br)cc1Cl c1(C(=O)NCC2N(C)CCN(c3snc(C(C)C)n3)C2)ccc(P(C)(C)=O)cc1 C#CCC(CC(F)F)C(=O)N1CCC(CCC(=O)NCCn2ccccc2=O)C1 C12COC(C)(C)CN1C(=O)N2.Cc1cc2sc(Sc3ccn(CCF)n3)nc2s1 c1(NC(C(CN(C)C)NC(c2cnc(C)n2C)=O)=O)ccc2c(c1)CCC2 C1(CNCc2cn(CC)nc2)CC(F)CN1C(c1ncc(F)cn1)=O CC(O)(CNC(c1csnc1C1CC1)=O)CNC(c1cnn(CCO)c1)=O c1(C(N(C=O)CC2N(C)CCC2)CF)ccc(C(F)(F)F)cc1 CCCC(C)(CO)NC(c1cc(-c2ccccc2Cl)c(C)s1)=O c1(CC(C(=O)NC(C(C)C)CNC(=O)C(=O)NCC(F)(F)F)O)ccc(Cl)cc1 Cc1cc(C(F)(F)F)nn1CC(=O)NCCO.n1(CCCC(=O)O)cc(CC(C)C)nn1 N1(C(c2c(C)nns2)=O)CCCCC2(CCN(C(=O)C(C3CCOCC3)O)C2)C1 n1(CC)cnc2c(NCc3cc(F)ccc3C)[nH]c(=NC(CCO)C(F)F)nc12 c1(CC(=O)NCC2CN(C3CC3)CC3(CCC3)O2)c[nH]c2ccc([N+](=O)[O-])cc12 CC1(C)COCC(C(=O)NCCCOCCNC(=O)CCc2cnn[nH]2)O1 C=C(Br)CN=C(NCC1CCCO1)N1CCCC(CC(C)(C)C(N)=O)C1 C(C(C)(C)CC(=O)NCC1CCCN1C(C)C(=O)NC)OC C1(CNC(CSC(C)C)=O)(CNC(c2cnn(CCF)c2)=O)CC12CCC2 C12(NC(C(CC=C)OC)=O)CCCC1N(C(c1cc(N(C)C)ccn1)=O)CCC2 N1(C(C(C(C)C)SCC)=O)CCC(CNC(C2(C3CCC3)CC2)=O)CC1C c1(NC(c2cnc(C#N)c(Cl)c2)=O)cnc2c(c1)CNCC2 C1(O)(CCNC(C2C(C)(C)CO2)=O)CCN(C(c2cncnc2)=O)CC1 c1(NC)cncnc1NC1CCCN1C(c1ccc(CC(C2CC2)C2CC2)cc1)=O C1(NC(=O)CC2CS(=O)(=O)C2)CC12CCOc1ccccc12 c1(CC)c(C(N2CCC(OCCNC(=O)C=CC3CC3)C2)=O)nnn1C C(=O)(C1CCCc2c1ncn2C)N1CCN(C(CC(C)C2CCCCC2)=O)CC1 c1(CNC2CC(C(=O)NC(c3nccn3C)CC)C2)ncccn1 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC2CC1CCC2NC(C12CC(C)(C1)C2)=O N1(C(C2CC(N(C)C)C2)=O)CCOC(CNC(C2CC(N3CCCC3)C2)=O)C1 C1(COC(C2(C(=O)OC)CCCCC2)=O)CC(c2ccc3c(c2)CCO3)=NO1 C1(NC(C(C)(F)F)=O)CCCN(C(=O)CC2=CCCCC2)CC1F C(=O)(CN=c1cc[nH]cc1)N1CCC(=C)CC1C(=O)NCC(F)C1CCC1 C1(N(C(=O)CN2CCCC2=O)CCC)CCN(C(=O)Cc2nocc2C)CC1 c1(C(=O)NC(C#C)CC)cc(CNC(c2cnsc2)=O)ccn1 C1(NC(C(CC)c2ccccc2)=O)COCCN(C(=O)Cn2ccnn2)C1 C1(NC(C(C)CC(N)=O)=O)CC2COCC(C1)C2NC(c1cc(Cl)c(Cl)n1C)=O C1(CNC(C(CCOC)NC(=O)COC(C)(C)C)=O)CC(C)OC(C)C1 C1(NC(C(CCC)O)=O)CC2CCC(C1F)N2C(=O)C(F)CCC(C)C C=CCN=C(NCC(c1cccc2ccccc12)O)N1CCC2CCCCC2C1 c1(SCC)cc(C(=O)NC2CCCC2NC(=O)CC2CC=CCC2)ccn1 C1(C(=O)NCCC2CCN(C(C(C)=C(C)C)=O)C2)CCCCS1(=O)=O CC1CCc2nc(C(=O)N(C3CN(C(C4SCCCS4)=O)CC3O)C)cn2C1 c1(CCNC(CCN(C(=O)Cc2ncoc2C)CC)=O)cn(C)cn1 C1(NC(CC(=O)OC)=O)CN(CC(=O)Cc2ncccc2C)CCC1C(F)(F)F N1(CC(N2CC(C(c3cn(CCCN(C)C)nn3)C)C2)=O)CC2CCC1C2 c1(NC(=O)Cc2ccc(Cl)cc2)cc(C(N2CCN(C)CC2)=O)c(N(C)C)cn1 CC(C)CC(C)(CN=c1ccnc[nH]1)NC(c1cccc2cccnc12)=O C1(NC(Cc2n(C)nnc2)=O)CC2CC(C1)N(C(c1cc(N)cc(O)c1)=O)C2 Cc1csc2c(N3CCC(C)C3CNC(c3cnc(N(C)C)cn3)=O)ncnc12 C(=O)(CC(=O)NC(CNC(C1(n2cccn2)CC1)=O)CCOC)NCC C(CC(O)CNC(c1cnn(CCC2CCCC2)c1)=O)NC(C1(N(C)C)CC1)=O Cc1cccc(Br)c1C(C(=O)NC1CC(=O)N(O)C1)NC(c1cc(C2CC2)no1)=O c1(C(=O)NCC(C)OCc2ccccn2)ccc(F)cn1 N1(C(=O)COc2ccccc2)CC(CO)C2(CCN(C(C3CC34CC4)=O)CC2)C1 c1(C(N2CC(CCNC(Cc3cn(C)nc3)=O)C2)=O)cnn2c1S(=O)(=O)NCC2 CCCCCCCCC(=O)NC1CN(C(=O)C(C)(C)CC(=O)OC)CC12CCC2 N1(C(C(CC)n2ccnc2)=O)CCC(O)C(NC(c2nn(C)nc2C)=O)C1 c1(C(=O)NC(C)C(C)NC(=O)CNS(=O)(=O)N(C)C)ccnc2ncsc12 c1(C(C)O)ccc(NC(=O)CC2CCN(C(c3cso3)=O)C2)cc1 c1(C(C(=O)NCCSC)N(C2CCCSC2)CC)ccc(F)c2ncccc12 CC1CN(C(c2cc[nH]n2)=O)CCC1NC(C1(C(F)F)CC(=O)C1)=O c1(CNC(=O)OC(C)(C)C)ncccc1C(=O)OCC(N1CCC1)C1CC1 CC(=O)CCCC(C)C(=O)N(C)CCNC(=O)Cc1ccon1 c1(C(=O)NC2(C(N(C3CC3(C)C)C)=O)CSC2)ncncc1N Cc1cc(C2CC2)ncc1C(N1CCCC(F)(CNC(c2ccoc2C)=O)C1)=O c1(C(C(F)(F)F)COc2ccc(OCC)cc2C(F)(F)F)ccc([N+](=O)[O-])cc1 C1(C(=O)N(C)CC2CCCC2(C)C)(CC)CCN(C(C2CC2(F)Cl)=O)CC1 C(CC(=O)NC1CCCC(C(N)=O)C1)(C(F)F)NC(CC1ON=C(CC)C1)=O N1(C(C(C)OC2CCCCC2)=O)CC2CC1C2NC(c1ccnnc1Cl)=O C(CC(C)C)(C(=O)Nc1cn(C)nc1C(N)=O)ONC(c1c(CCC)[nH]cc1)=O CN1CCN(CC(=O)NCc2ccccc2CNc2cc(=O)n(C)cn2)CC1=O c1(C(=O)OC)nsc(=NC(C)C2CCCN(C(=O)C(N3CCSCC3)C)C2)[nH]1 C1(CC)CCN(C(c2ccccc2C)=O)C1C(=O)NCC(C)(C)CCOC c1(C(=O)OC)ccc(N2CC3CC3(C(=O)NC3CCC(F)(F)C3)C2)c([N+](=O)[O-])c1 CCCC(C(=O)OC)C(=O)N1CC(F)(F)CC1CNC(c1c(C)cnn1C)=O C(=O)(CCCC(CC)CC)N1C(C(=O)NCC(CC=C)(F)F)CC1C C=CCCC(O)CN(C(=O)CC1CCN(C(c2ccccc2)=O)C1)C C1(C(=O)NCC2CCC3(CC3)C2)CCN(C(=O)Cn2cnnc2)C12CC2 C(=O)(CCCN(C)N=O)NCCC1(O)CN(C(C(C)(C)NC(=O)OC)=O)C1 c1(C(=O)NCCN(C(c2csc(CN(C)C)c2)=O)CC)cnc(SC)n1C N1(c2nc(C)nc(C)c2F)CC2C3CCC(C2C1)N(C(=O)CC1=NNC(=O)C1)C3 c1(OCC)nc(C(=O)NC2CC(C)N(C(=O)C=C(C)C)C2)cc2ccccc12 CC(C)CC(CNC(c1cc(CO)on1)=O)C(=O)NCCN1CCCCC1C C1(CNC(c2c(C)cco2)=O)CC(NC(c2cc(C(F)F)cs2)=O)C(O)C1 C1(CNC(C2C(CC(C)C)C2)=O)CCN(C(=O)C2=NOCC2)CC1O C(C)(C(C)NC(=O)CCc1nc[nH]n1)NC(COCC(=C)C)=O S(=O)(=O)(CCN1CCc2cccnc21)N1CC(C(=O)O)OCC1 C=CC1(CC(=O)N(CCCOCC(C)C)C2CC2)CN(C(=O)Cc2ccoc2)C1 c1(OC)cc(CN2CC(C(N3CCC(O)C3)=O)CC(F)C2)ccc1C(F)(F)F c1(C(N2CCC(C)(NC(=O)CC3CCCO3)CC2)=O)ccc(F)c(F)c1F c1(C(=O)NC2C(NC(C(C)CN3CCOCC3)=O)C2)cc([N+](=O)[O-])ccc1Cl Cc1cc2c(C(=O)NCCCC(C)NC(=O)CCC3CC3C)ccc(C)c2[nH]1 CCC(C)(CO)C(=O)NC1CC(Nc2cnc(F)cc2C)C1 CCCCC(C)CCC(=O)N1CC(OCCC(N2CCC3CC23)=O)C1 N1(C(C(CCSC)NC(c2c[nH]c(C)c2)=O)=O)C2C=CCC1CCC2 N1(C(c2c(C)ccs2)=O)CCC2C(C1)NC(=O)CN2C(=O)C1=CC(C)CC1 Cc1cc(=NCCCNC(c2ccccc2)=O)[nH]c(=NCC23CCN(CC2)C3)[nH]1 c1(C(n2nnnc2N2CCOC(C3CCOCC3)C2)C)cc(S(N)(=O)=O)co1 c1(C(N(CC(CC)NC(=O)CC(C)C)CC)=O)ccnn1COC c1(C(N2CC(CNC(=O)CCCF)CC(C)C2)=O)ccc2ccncc2c1 N1(C(CNC(C)=O)=O)CC2CC1C2NC(C1CC1c1ccnn1C)=O C#CCN(OC)C(=O)C1(F)CCNC1.C(=O)(C(CC)C(=O)OC)NC CC1(C(F)F)CN(CC(=O)N2CCC2)CCO1.c1(CN)ccc(OCC(F)(F)F)nc1 CCCC(C(=O)NCCOCCOCCNC(=O)CCCC(F)(F)CO)C(C)C NC1C2CC3C(C2)C13CN1CCCCC1c1nccs1 C12(NC(C3(C4CC4)CN(C(CC(C)F)=O)C3)=O)CC3CC(CC1C3)C2 c1(C(=O)NC(CC)CNC(c2ccc(C(C)C)c(Cl)c2)=O)cc2c(ncn2C)s1 C(=O)(C(C(C)CC)C1CC1)N1CC(C=C)(CC(=O)NCCCCCCO)C1 Cc1ccc(C(=O)NCC(C)N(C)C(C2NC(=O)OC2C)=O)cc1C C1(C)(CC)CC(NC(c2cnn(C(F)F)c2)=O)CN1C(c1cccc(=O)o1)=O N1(C(C2CC(CC)C2)=O)CC(C)OC2(CCN(c3ncnc4[nH]ccc34)CC2)C1 c1(CC(=O)NCC=CCNC(C2(CC#C)CC=CCC2)=O)ccc2c(c1)OCO2 c1(C(=O)NCC2C(C)(C)CN(C(=O)CC3CCC(=O)N3)C2)cc2ccccc2o1 N1(C(C(COC)(C)C)=O)CCN(C(c2ccc(C(F)F)c(F)c2)=O)CC12CCC2 CCC(CC1CCCC1)C(=O)NCC1(F)CC(NC(C2(CO)CC2)=O)C1 C(=O)(C1=CS(=O)CCC1)OC1CCCN(C(C)(C)Cn2cc3c(n2)CCCC3)C1=O Cc1cccc(C(=O)NC2(CCC(=O)N(C)CC3CC3C)CCCC2)c1F c1(C(N2C(CNC(C3(C)CC3)=O)CC(C(F)(F)F)C2)=O)cc(O)ncc1Br C1(C(=O)NCC(C#C)C(C)C)CCN(C(=O)C=Cc2cncn2C)C(C)(C)C1 C1(CC)C(C(=O)NCC(C)CN(C(=O)CCSC(F)(F)F)C)CCN1C c1(C(=O)NC2CN(C(CCOCCOC)=O)CC2O)cc(S(N)(=O)=O)co1 c1(CC)ccc(-n2nc(-c3ccc(N)cn3)nc2C(c2ccc(Cl)cc2)C)cc1 c1(CNC(C2N(C(COC(C)=O)=O)CCC2)=O)cnc2cc(C)ccn12 c1(C(=O)NC(CC)CN(C(=O)C(CC)N(C)C)C)cnc2n1CCCCC2 C1(C(=O)NC(CCC)C2CCCC2)CSCCN1C(=O)Cc1ccc[nH]1 C1(COC)CN(C(c2cnn(C)c2Cl)=O)CCN1C(=O)CC1CCC(F)(F)C1 c1(C(=O)NC2CCN(C(C(CC)(C)C)=O)C2)cc(F)c(F)cc1I C1(C(=O)Nc2c(N(C)C)cccc2)CCCN(C(c2cn(C)ccc2=O)=O)CC1 Cc1ncc(C(N2CCC2CNC(c2ocnc2C(F)(F)F)=O)=O)n1C N1(C(CCCC#C)=O)Cc2ccccc2C(CNC(c2cn(CC)nn2)=O)C1 N1(C(C2CCC(C)O2)=O)CC2C(CNC(=O)CC(C)(F)F)C2C1 S(=O)(=O)(c1ccccc1[N+](=O)[O-])N1CCN(CC(CC)(C)CO)CC1 C(CC(F)F)(C(=O)N1CCC(O)CC1C)NC(c1scc(C)c1)=O c1(C(=O)NC2(C)CCN(C(C3CCCC(C)C3)=O)C2)ccn(O)c(=O)c1 c1(NCCNC2(S(C)(=O)=O)CCC2)nc2ccc(F)cc2c(=NC2CCCC2)[nH]1 Cc1cn(CC(N2CCC3CN(C(=O)CSC(F)F)CC23)=O)c(=O)nc1O Cc1ccc(SCCNC2CCCCC2c2ccc(F)cc2)cc1 C1(C(=O)NCC(COCC)C)(NC(c2cn(CC)nc2C)=O)CCOCC1 C(C(=O)NCC(C)N(C)C(c1sccc1-n1cnnn1)=O)(C(C)C)OCC(C)C C1(CC(N2C(Cn3cc(CN(C(C)C)C)nn3)CCC2)=O)CCC(C)(C)CO1 c1(C(N(C2CCN(C(c3cccn3C)=O)C2)CC)=O)ccn2ncnc2c1 c1(C(C)OC(=O)CSc2ccccc2)cccc(S(=O)(=O)N(C)CCN)c1 C(CCCCCO)Cc1cn(C2CN(C(c3sccc3F)=O)C2)nc1 CC1CCN(C(=O)C2=COCCO2)CCN1C(=O)Cc1cncn1C N1(C(c2c(C)nccn2)=O)CCC2(CN2C(=O)CCc2cc3ccccc3o2)C1 N1(C(c2c(C)cnnc2)=O)CCC(C(N2CC(c3ncc[nH]3)C2)=O)C12CC2 CCC(COC)C(=O)NCC(C)CN(C)C(C1COC(=O)N1)=O C1(NC(c2cc(C(C)C)on2)=O)CC2CC(NC(C3(F)CC3C)=O)C1C2 N1(C(C=CCC(C)(C)NC(C2COC(=O)N2)=O)=O)Cc2ncsc2C1 N1(C(CCN(C(=O)CC2COCC(C)O2)C(C)C)=O)C2CCC1CN(C)C2 C=CC(C)(CC)C(=O)N1CC(NC(C2(N3CCOCC3)CCCCC2)=O)C(O)C1 CC(C)C(C(=O)N1CC2CC1C1CC21)C(C)NC(c1ccc(F)c(F)c1)=O C1(CNC(Cc2cnc(C)o2)=O)CC(NC(=O)CCc2csc(C)n2)CC1O c1(-c2cc(C(N3CC(CNC(CC=CC)=O)C3)=O)no2)ccccc1[N+](=O)[O-] n1(CC(=O)NCCN(CCC)C(c2nc(-c3ccccc3)no2)C)cc(Cl)cn1 C1(CCNC(C(n2ccc(C)n2)C)=O)CC(F)(F)CN1C(c1nnccc1C)=O c1(CCC(=O)N(CCCOC)CCO)nccn1C C=CC1(C(=O)N(CC(=O)NC(C)(C)C)C)CCN(C(=O)C2=CCCOCC2)CC1 C(=O)(C1=CC2CCCCCC12)N1C(CNC(C(c2ccccc2)C)=O)CCCC1 CC1=C(C(=O)NC2CN(C(C3(O)CCCC(C)(C)CC3)=O)C2)C(=O)OC1(C)C c1(OC)c(C(N2CCC(O)(CNC(C3CCC(=O)N3)=O)C2)=O)cc(Cl)cc1C C1(C(c2cn(CC3CCCO3)nn2)NC(N)=O)CCCCN(C(=O)CCc2cncs2)C1 C1(CCC#C)CCCN(C(=O)C(C)C(C)NC(=O)Cn2c(O)nnc2O)C1 CC1CC(CNC(=O)CCc2ccc[nH]2)CN1C(=O)CCC1CC1(C)C c1(C(=O)NC2CCC(CNC(c3[nH]cc(C)c3)=O)C2)cnc2cc(C)nn2c1C C(C(=O)N1CCN(C(=O)C(C)(O)C2CCCC2)CC1)(C(C)(C)C)c1n(C)cnn1 c1(C(=O)NC(C(=O)NC(CCCC)COC)Cc2ccoc2)occ2c1CCC2 c1(C(=O)NC2CC(N(C(=O)Cn3ccc(C4CC4)n3)C)C2)[nH]nc2c1CCC2(C)C Cc1ncc(Cl)cc1CC(N1CCCC(N(CCF)C(c2cnsc2)=O)C1)=O c1(CC(C)NC(c2c(C)[nH]nc2CO)=O)ccc(C#N)cc1F CCS(=O)(=O)c1cccc(CC(=O)NC2CC(NC(=O)Cc3ccnn3C)C2)c1 C1(NC(c2ccc(O)o2)=O)CC2CCC(C1)N2C(c1ccnn1C(F)F)=O c1(C(N(CC(CN(C(C(C)(C)OC)=O)C)O)C)=O)cc(N)c2ccccc2n1 C1(C(=O)NCc2c(C)n[nH]c2)CCN(C(c2ccc(CF)cc2)=O)C1C N1(C(CSCCC)=O)CCCC(NC(c2sc(F)cc2Cl)=O)C(F)C1 N1(C(C2CCC(OC)C2)=O)CC2CCC(N(C)C(C3CCCS3)=O)C2C1 Cc1cc(C)n(CC(=O)NC(C)CN(C(=O)Cc2csc(Cl)n2)C)n1 C(=O)(CCS(=O)(=O)N1CCOCC1)NC1(CC)CN(C(c2ccc(Cl)cc2)=O)C1 Cc1nc(N2CCC(C)(CNC(=O)C=CC3CCCO3)CC2)c2c[nH]nc2n1 c1(C(=O)NCC2(OCC)CCN(C(C3(CC=C)CC3)=O)C2)cc(C)nc(O)n1 C1(C(N2C(CO)CC(OC)C2)=O)CNC(=O)CN1C(=O)C=CC1CCC1 C1(C(C(=O)OC(C(C)=O)C)O)CCN(C2CCC2)CC1 C1(NC2CCN(C)CC2c2ccnn2C)C2Cc3ccc(Br)cc3C12 C(c1ccoc1)=CC(=O)NCC(CO)NC(c1occc1Cl)=O C1(NC(c2c(Cl)ncc(C)c2)=O)CN(C(=O)Cc2cnn(C)c2)C2CCCCC12 N1(C(CCC(=C)C)=O)CCC(NC(c2cc(Br)cn2C)=O)C(CC)C1 C1(NC(C2(COC)CC2)=O)CCC(O)CN(C(=O)CCN2C(=O)CCC2=O)C1 n1(CC(CC)C)cc(CNC(=O)Cn2cnnc2)nn1.C1C(=O)O1 c1(C(=O)NCC2C(NC(C3=C(C)CCC3)=O)C2)cc2cc(F)c(F)cc2[nH]1 c1(C(=O)NC(CC)CN(C(=O)CC(C)(C)SC)C)cc(Cl)cc(Cl)c1 n1(CC#C)cnnc1C(N1CCC(N(C(=O)C(CC)NC(=O)OC)CCO)C1)=O N1(C(c2cc(C)n(C(C)C)n2)=O)CC2CC(CNC(C3CCCN3C)=O)C2C1 c1(C(=O)NCC2(F)CCC(NC(CCCC)=O)C2)cc(F)c(CC)cc1F c1(C(=O)NC(C(=O)NC(C(=O)NC(C)C)C)c2ccoc2)ccoc1Cl CC(C)(CC(F)C(=O)NCC1CC1(F)F)NC(c1cnc[nH]c1=N)=O Cc1ncc(C(=O)NC2(C)CCN(C(=O)CCc3cccc(O)c3)CC2)c(C)n1 N1(C(C2(C(C)(F)F)CC2)=O)CC=CC1C(=O)NC1(C(=O)N(C)C)CCCC1 c1(C(=O)NCC2C(NC(c3csc(CO)n3)=O)CC2)cc([N+](=O)[O-])n[nH]1 c1(C(N(C)Cc2c(CNC(CCCCOC)=O)cccc2)=O)ccc(F)cc1C n1(CC(=O)NCCCN(C(=O)CCc2cncn2C)CC)ncc(Br)n1 c1(C(=O)NCCCN(C(=O)C(CCSC)OC)CC)nc(C(F)(F)F)ccc1F N1(C(CCC#C)=O)CCC2CCC(NC(C3CC34CCOC4)=O)C1C2 CCC(C)(CNC(=O)C(C)Oc1ccccc1)NC(=O)CC1CSCCO1 N1(C(C(COC)(F)F)=O)CCC(CO)(CNC(c2ccc(C#N)cn2)=O)CC1 CN1CC(O)CC1CNC(C1(C2CCCN2C(=O)C)CC1)=O.C1(O)CC(F)(F)C1 N1(C(C2C(C)OC(C)C2)=O)CC(CO)C2(CCN(C(C3(C(F)F)CC3)=O)CC2)C1 Cc1cc(C)c(C(N2CCC(NC(c3sccc3C)=O)C(O)C2)=O)c(O)n1 C1(C)(C(=O)NCCCN(C(C2C(C)CCC2)=O)C2CC2)CCC(C)(C)CC1 c1(C(=O)NC2(CNC(c3n(CC(C)C)ncc3)=O)CC2)csc2cncn12 CCCCC(C)C(=O)NCCN(C(=O)COc1nnc(S)n1C)CCOCC C1(C)(C(=O)NCC(C)NC(C(c2cncc(F)c2)C)=O)CCC2CC2C1 c1(C(N2CCC3C(NC(CC(CC)(C)C)=O)C32)=O)cc(N)c2ncccc2c1 CC(C)CC(C)(O)C(=O)N(C)CC1CCC(NC(=O)CCc2ncc[nH]2)CC1 Cc1nc(C)c(C(=O)NC2CN(C(=O)CCC3CCCC3)CC2C)c(C)n1 N1(C(=O)CCc2cncs2)CC2CN(C(=O)CSCc3cscn3)CC2C1 Cc1c(Cl)ccnc1C(=O)NCC(O)CN(C(=O)Cc1coc(C(F)F)n1)C c1(CN=[N+]=[N-])ccccc1C(N1CC(N2CCN(C(=O)Cn3nccn3)CC2)C1)=O C1(C(=O)OC)CN(C(C2CCC2(C)C)=O)CCC1(C)C C(CN=c1ccc(Br)c(S(=O)(=O)N2CCC(n3cncn3)C2)[nH]1)OCCSC N1(C(C(C)OC)=O)CC2(CCOCC2)CC1CNC(=O)C=Cc1ccccn1 N1(C(CCCC(C)=O)=O)CCC2(CC1)CC(C)N(C(=O)CCc1cnn(C)n1)C2 N1(C(CCC(CC)NC(c2ccc(C)nn2)=O)=O)CC2(CCN(C)CC2)C1 N1(C(c2ccc(OCC)cc2)=O)CCN(C(=O)C(C)CC(C)C)C(CO)C1 c1(C(=O)NCC(CNC(CCc2nc(C)sc2)=O)O)cc(Cl)c(F)cc1O C#Cc1cncc(C(N2CCN(C(=O)C(C)n3cncn3)CC2CO)=O)c1 N1(C(C(C)OCC2CC2)=O)CC(O)(CN(C(=O)Cc2csc(C(C)(C)C)n2)C)C1 C#Cc1cc(C(=O)NC2(CC(=O)NCC3=CCN(C(C)=O)CC3)CC2)ccc1C Cc1cccc(NC(C2CCC(NC(C3(Br)CCC3)=O)C2)=O)n1 C1(CC(C)NC(CCC=C)=O)CCN(C(=O)CCOCCOC)CC1 CC1(CNC(=O)C(F)F)CCN(C(=O)Cc2ccon2)CC1 Cc1nc(-c2c[nH]cc2C(=O)NC2CC(C(C)=O)C2)cs1 C1(NC(c2c(C)noc2)=O)CCN(C(c2cc(C3CCCC3)[nH]n2)=O)CC1F C(CC(C)C(=O)NC(C1CC1C(=O)NCC12CC(F)(C1)C2)C)OC C1(C(=O)NCC2(F)CN(C(=O)C(c3ccccc3)=O)C2)C(F)(F)C12CC2 C12(NC(c3c(C)nc(C)s3)=O)CCOC(CNC(=O)Cc3cncn3C)(C1)C2 C1(O)(CNC(c2cnc(COC)s2)=O)CCN(C(C2CC(=O)NC2(C)C)=O)CC1 c1(CC)cc(C(N2CCC(C)(NC(c3ccc(OC)o3)=O)C2)=O)cc2c[nH]nc12 c1(C(=O)NCC(C)NC(=O)C(F)(F)C(O)C(C)C)cnc2c(c1)nc(O)n2C C(=O)(C(C)(C)C(F)c1ccccc1)N(CCNC(c1cn(C)c(O)n1)=O)CC1CC1 C1(CC(N2CC(C)C(CC(=O)NCc3nc(=O)n(C)[nH]3)C2)=O)CCC2(CC2)CO1 C1(NC(C2=CCC(C)C2)=O)C(C)CN(C(c2ccncc2C(F)(F)F)=O)CC1C C1(C2(C)CC2)COCCN1C(=O)C(CNC(c1cocc1C(N)=O)=O)CC1CC1 c1(C(=O)OC)cc(Br)c(C)cc1NC(=O)C(=O)NCC(c1ccc(F)cc1)(C)C CC1(C)CCCC1C(=O)NCC1(F)CC(NC(c2cccn2C2CC2)=O)C1 C12(C(=O)NC3CCC(CNC(c4cc(C(=O)OC)sc4)=O)C3)CCCC1CCC2 C(=O)(C(C)(C)S(C)(=O)=O)NC1CCCC(CN(C(C2(C=C)CCCCC2)=O)C)C1 C1(NC(c2n[nH]cc2F)=O)CCCN(C(C2(F)CC2)=O)CC1 C1(C(=O)NC2CC(CNC(c3cccn3-c3ccccc3)=O)C2)(CC)CCOC1 C(CCC(C)(C)C(=O)NCCCC1CC1C)NC(Cc1scc(C)c1)=O C1(CC(N2CCC(CNC(c3c(CC)ncs3)=O)C2)=O)CC(C)(C)CO1 C1(C(=O)NCC(C2CCCC2)C)CC(F)(F)CN1C(C1CC(F)CN1C)=O C(=O)C1Cc2ccccc21.C(=O)(C1=CCCN(C)C1)N1CCC(OC)C1C C1(C)(CNC(CCCC#C)=O)CN(C(c2cc3sccc3s2)=O)CC1C N1(C(C)=O)CCC(N(C(=O)C(CCN(C)C)NC(C2(C)CCOC2)=O)C)CC1 CCC(C(=O)NC1CC(CC(=O)NNC=O)C1)OC.C1(C)CCCC1CCO C1(C)(CNC(CCSCCCC)=O)CCCN(C(=O)C(C)C(=O)OC)C1 c1(CN2CCC(NC(=O)Cc3c(Cl)cccc3Cl)C(F)C2)c(Br)cc(F)c(F)c1F c1(N(CC(N2C3CSCC2C3)=O)Cc2cccnc2)ncc(Cl)cc1F C(=O)(C(C)CS(C)(=O)=O)N1CCC(O)(CNC(C2(CCC=C)CCCC2)=O)C1 c1(C(=O)NC2C(NC(C=CC)=O)CC2)ccc2n[nH]cc2c1C C1(C(=O)NC23CC(CNC(CNC(CCC)=O)=O)(C2)C3)C2CCOCC12 c1(CS(=O)(=O)Nc2c(C(=O)Nc3c(C)ccnc3)scc2)ccc(F)cc1Cl c1(C(N2CCN(C(c3cc(CC)on3)=O)C(C)C2)=O)cc(C)nc2[nH]nc(C)c12 C(CC(F)(F)F)(C(=O)N(C(C)C(=O)NO)c1cn(-c2cccnc2Cl)nn1)OC c1(C(=O)NCCCN(C(C(CC#C)C2CC2)=O)C(C)C)ccn2cccc2c1 C(C(C(=O)NCCCC1CC1C)C(C)(C)C)NC(CC(C(=C)C)OCC)=O N1(C(c2c(C)nc(O)cc2)=O)CC2CC(C1)CN(C(c1cnnn1C)=O)C2 N1(C(C(C)C(F)F)=O)CC=C(C(C)(C)C(=O)NC2CC(=C3CC3)C2)C1 C(=O)(C(CCO)C1CC1)NC(C1(CNC(=O)COCCCF)CC1)C c1(C(=O)N)cccc2cc(Br)cnc12.n12cc(nn1)C2(C12CC(CO1)C2)C.C1CC1 C1(CNC(c2[nH]cc(C(C(C)C)=O)c2)=O)CCN(C(=O)C(=O)N(C)C)C(C)C1 N1(Cc2nc(OC)nc(C)c2)CC(CO)CC12CCOCC2 C1(CNC(c2ccc3snnc3c2)=O)CC2(CCC2)CN1C(=O)COCC(F)F C1(C(=O)NCCCOCCCN(C)C)COC(C(F)F)C1.C1(=O)CN1 Cc1noc(C)c1CNC(N1CCCC1CN(C)C(=O)OC(C)(C)C)=O C1(NC(C)=O)CC(c2ccc(Br)cc2)N(C(C2CCCOC2C)=O)C1 N1(C(NC2CCn3nncc32)=O)C2CCC1CC(O)C2 C1(CNC(C2CCCS2)=O)CCCN(C(=O)C(C2CCCCC2)O)CC1 C(=O)(C1=NNC(=O)C1)N(C1CN(C(c2cn(C(C)(C)C)cn2)=O)C1)C N1(C(COc2ccn(C)n2)=O)CC(CNC(C2CCC3(CC3)C2)=O)CC1(C)C n1(CC)cc([N+](=O)[O-])c(C(N2CCC(F)(CNC(C3CCOC3(C)C)=O)C2)=O)n1 C12(NC(=O)NCC(CCC)C)CCCCC(C(=O)OC(C)(C)C)(C1)C2 N1(C(C2CCC(CCC)CC2)=O)CCC(NC(=O)COCC(F)F)C(CO)C1 N1(C(C)C)CCCC(CC(N2CCCC2CNC(=O)C(C)C#N)=O)C1 N1(C(CN(C2CCC2)C)=O)CCCCC1C1CCCN1C(=O)C=C1CCN(C)C1 C1(C(=O)NCC(CN(C(c2cc(CC)ncn2)=O)C)(C)C)CC2CCC1CC2 C1(C(N2CC(c3ccc(N(C)C)cc3)C2)=O)CCN(C=O)CC1O.C(C)(C)C#N n1(CC(=O)NC2C(NC(C=C(CCC)C)=O)CCCC2)ccc([N+](=O)[O-])n1 c1(NC(c2ccc(NC(c3c(I)ccnc3F)=O)cn2)=O)ccc(Cl)c(Cl)c1I CCC(CC(=O)NCc1ccccc1Cl)NC(=O)CCc1cc(C)no1 C1(CC)CN(C(=O)C(N2CCC(O)(C(F)(F)F)CC2)=O)CCC1C(=O)OC(C)(C)C C12(CNC(C(C3CCCCC3)OC)=O)CC1CN(C(C1CC(OC)C1)=O)C2 C12(C(=O)NCC(CNC(=O)CC3(n4cccn4)CC3)F)CCC(O)(CC1)CC2 N1(C2C(=O)NC3C2C3)CCNC(=O)C1.c1(C(NOCCCC#C)=O)cc(C#C)co1 c1(CNC(C2CC(C(=O)OC)C2)=O)cccc(Cl)c1F.C12(CC1)C(=O)N2 CCC(CC)C(C)C(=O)NCC1(OC)CN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1 C1(CNC(=O)CC2CC3(CC3)CO2)CCCCCN1C(=O)C(Cl)=CCl O=C(CCC(=O)c1ccccn1)NCCN(C(=O)C=Cc1ncco1)CC1CC1 C(=O)(CCCC(=O)N1CCOCC(NC(=O)C(CC)n2cccn2)C1)OCC C(C(C)(C)C#CC(=O)NC(C)CCn1cncn1)NC(C(C1CC1)SC)=O C1(C(N(CC)Cc2cc[nH]n2)=O)COCCN(C(C2CN3CCC2CC3)=O)C1 N1(C(CN2CC(C)(OC)C2)=O)C2CCC1CC(NC(C1CCCC1C1CC1)=O)C2 N1(C(C(CC)O)=O)CCC2CN(C(c3ccc(OC)nc3)=O)CC2CC1 c1(C(=O)NCC2C(CNC(C3(C)CCCCCC3)=O)C2)c(N)sc2c1CCSC2 C(=O)(CCCCC#N)NCC(CNC(CC(CC)C)=O)OC C(=O)(C#CC1CCOC1)NC1CC(C(N2CC(C#N)(F)C2)=O)OCC1 C(C(F)(F)CC(O)CO)NC(COc1cccc(-c2scc(C)n2)c1)=O N1(C(C2C(C)OCCC2)=O)CCCN(C(=O)C(C)(C)C2CCOCC2)CC1 c1(OCC(N2C(CCCNC(C(CC)F)=O)CCC2)=O)ccc(F)cc1CO CON1CCC(C(N2CC(NC(=O)C3=CCCSC3)CC2C)=O)CC1 C1(CC(=O)NCC(CC2CCCC2)C(=O)NCC(F)Cl)CCCC12CC2 C1(C(=O)NCC(CNC(c2csc(=N)[nH]2)=O)OC)CCC2(CCCC2)CC1 C1(C(=O)Nc2c(CC)nsc2)CN(C(C2(O)CCCCCC2)=O)CC12CC2 c1(OC)ccc(C)cc1CC(N1CCCC(C)C1CNC(c1cc(F)c[nH]1)=O)=O c1(C(=O)NCC2CC(NC(c3n(C)ccc3)=O)C2(C)C)cc2n(n1)CCC2 C1(C(=O)NCCOCCC#C)C2CCN(C(=O)CC(C)(C)C#N)CC12 C(C(CO)C(C)(C)C)NC(CC1CC(CC)C1)=O.C1C(=O)NCCS1 N1(c2cc(C)ncn2)CCN(CC(=O)Nc2cnc(Cl)c(Cl)c2)CC1C c1(C(=O)NC2CC(CNC(C(CC)C(C)O)=O)C2)sc2cc(OC)ccc2c1Cl c1(C(=O)NCC2(C)CC(NC(=O)COC3CCOC3)C2)cc(F)c(F)cc1N c1(N2CCC(C(=O)NC3(CCC)CC3)C2)nc(CN(C)C)nc2ccccc12 C1(F)(C(N2CC(NC(c3ccc(C)n3C)=O)C2)=O)CC12CCCCC2 c1(N2CCN(CC3CN(CCOC)C3)CC2)nc(C(N)=O)c2ccsc2n1 N1(C(C(CC#C)NC(c2cc(Cl)cn2C)=O)=O)CCCCCCC1 CC1(C)CCN(C(c2ncccc2N)=O)CC1C(N1CCC(F)(F)C(F)C1)=O C(C)(C)(CC(=O)N1CCCCC1CCC(=O)NCCCc1cnccn1)N(C)C C1(N(C(=O)COCC(=O)OCC)CCC)CCNC2(CCC2)C1 c1(C(N2CCC(C3CCCO3)C2)C(=O)NC)ccc2c(c1)sc(=O)n2C N1(C(COc2c(C)ccc(C)c2)=O)CC(NC(=O)CCC(F)(F)F)C(C2CC2)C1 Cc1ccc(Oc2cncc(C(=O)NC3CC(NC(=O)OC(C)(C)C)C3)n2)cc1 c1(CC(N2CC(CC)C(NC(c3cnco3)=O)C2)=O)cccc(F)c1Br C1(NC(C2(CC)CCOC2)=O)CCN(C(=O)Cc2csc(C)n2)CC1C N1(C(C(C)Cn2cccn2)=O)CCC(CN(C2(CO)CC2)Cc2cn[nH]c2)CC1 c1(C(=O)NC(CC=C)CNC(=O)C(F)=C(C)C)sc(S(N)(=O)=O)cc1C N1(C(C(C)NC(=O)OC)=O)CC2CCCC(NC(c3coc(Cl)c3)=O)C2C1 C1(NC(C(CC)OCC)=O)CCN(C(C2CC(C)=NO2)=O)C(C)C1 CON(CCC(=O)NC1CC1)C(=O)C(C)CC=C(C)C.C1COC(=O)N1 N1(c2ccnc(CC)n2)CCC(NC(=O)C(CO)NC(N)=O)C2(CCC2)C1 C(=O)(C(C)(C)CC(F)(F)F)NCC1(C)CCCC1NC(C1CCC2(CCC2)O1)=O CC1CCC(NC(=O)CCC2CC2(Cl)Cl)CN1C(=O)Cc1c(Cl)cnn1C CC1(C)CC2(CC2C(=O)NC(C2CCCN2C(=O)Cc2cccnc2O)(C)C)C1 C=CCC(CC=C)C(=O)N(C(C)CC(=O)NCC1CCC2(CC1)CC2)C C(CCCC(=O)N(CC(O)CN(C)C(C1CCCC(C(N)=O)C1)=O)C)OCC N1(C(CCOCCC)=O)CC(C(N2CC(=O)NCC2C)=O)CC(C)(C)C1 CCCC(=O)NCCC(C)NC(=O)CCc1cnco1 C1(CNC(c2ccc(C#C)o2)=O)CC(F)(F)CN1C(=O)CC1(OC)CCCC1 N1(C(N2CC(N3CC4CCC3C4)C2)=O)CCN(C(c2ccc(Br)cc2)=O)CC1 C(=O)(CC(C)(C)O)OCCN(C)Cc1cn(C(C(=O)OCC)(C)O)nn1 C1(NC(COCCC)=O)CN(C(c2cccnc2-n2cncn2)=O)CC2CC12 C1(CC=C)(NC(=O)CN2CCOC(C)C2)CCN(C(C2(CC)CC2)=O)C1 C1(C(=O)NC2(CC=C)CN(C(=O)CSc3ccccc3)C2)CC12CCSCC2 Cc1ccc(C(N2CC(OCC(=O)NCC(C)(C)C)C2)=O)c(F)c1 c1(CNc2c(C)c(NC3CCN(C4CCC4)CC3)ncn2)ccc2c(c1)CCC2 c1(CC(N2CCC(c3ccon3)CC2)=O)nc2ccc(C(F)(F)F)cc2s1 NS(=O)(=O)CCCC(=O)NCC(F)CNC(c1cnn(C2CCOC2)n1)=O S(=O)(=O)(c1cccs1)NCC(=O)N(C)C.C12CC(=O)N(C1)Cc1cn2nn1 c1(-c2cn(C3CN(C(CSS(C)(=O)=O)=O)C3)nn2)ccc(OCC(F)(F)F)cc1 N1(C(c2c(C)scc2)=O)CCCC(F)(C(=O)NCC(C)(C)C#N)C1 Cc1cc(NCC=CCNC(C2Cc3ccncc3C2)=O)ncc1[N+](=O)[O-] C1(C(=O)NCC2N(C(CCOCCOCC)=O)CCOC2)CCc2c[nH]nc2C1 c1(C(N(C)CC2CCCN(C(C3(OC)CC3)=O)C2)=O)cnc2ccccc2c1 C1(C(N2CC3CC3C2)=O)CC(NC(CCN(CC)CC)=O)C1(C)C N1(C(C(CCC)C(C)C)=O)CCOC2(C1)CN(C(C1CN3CCCC3CO1)=O)C2 c1(C(N(C2CCN(C(c3cc(OC)c(C)cc3)=O)C2)C)=O)cc(Cl)cc(C)c1N N1(C(C(CC)Cl)=O)CCC2(CCC2)C(CNC(=O)CC=C(Cl)Cl)C1 c1(C(C)C)nn(C)cc1C(c1nnnn1C(C)C)C(C)(C)C.C(CCCSCC)N c1(NC)ccc(S(=O)(=O)N(C(C)CCOC(C2CCCOC2)=O)C)cc1COC C1(C(=O)NCCS(=O)(=O)NC)N(C(=O)Cc2c(C)noc2Cl)CCCC1(C)C c1(OC(C)C)ccc(C(=O)NCCC(O)CNC(=O)CCn2ccnn2)nn1 CC1(C)C2CCC1(C(=O)NC1CCC3CC1CN3C(C13CC1C3)=O)CC2 CC(C)C(CO)CCNC(=O)CC1(NC(=O)C(C)CCN(C)C)CCC1 c1(C(=O)NC(C2CCN(C(C3CC(C)(C)C3)=O)C2)C)nc(C(F)(F)F)cs1 CC1(C)CC(C)(C(=O)NCCC2CSCCN2C(C2CCCCS2)=O)C1 c1(CC(C)C)ccc(NC(C2CCCC(NCc3nccn3C)C2)=O)cc1 C1(CNC(=O)C=CC2CCCC2)CCCCN(C(=O)C=CC2CCCO2)C1 C(=O)(CCC(C)NC(C1CN(C(C)C)C1)=O)NC(CCC=C)C1CC1 C1(CCC)(C(=O)NCC2(CNC(c3cscc3C)=O)CC2)CCNC1=O CCCCCCC(C)(C)C(=O)NC(C1CCCN1C(c1cnn(C(C)C)n1)=O)C C1(NC(=O)Cc2cc(Cl)sc2Cl)CCCN(C(=O)C=Cc2ccncn2)CC1F C(C)(C)(CC(=O)N1CCC(N2CCN(C(=O)COCC(F)F)CC2)C1)OC C1(NC(C(CN(C)C)NC(CC2(CSC)CC2)=O)=O)CC1C1CC1C C1(CNC(C=CC(=O)N(C)C)=O)CC2CCC1N(C(=O)CCCNS(C)(=O)=O)C2 CCCS(=O)(=O)C(C)C(=O)N1CCN(CC2CN(C(=O)CSC(F)F)C2)CC1 N1(C(CCOCC(C)(C)C)=O)CC(NC(c2nc(Cl)sc2Cl)=O)CC(O)C1 c1(C(=O)NC2CC(CNC(c3ccc(CCC)cc3)=O)C2)cnn2cccnc12 c1(CC)cc(C)c(C(N2CCC(O)(CCNC(=O)Cc3cc(Cl)n(C)n3)C2)=O)o1 c1(NC(C2(C#C)CC2)=O)cc(CC)cc(O)c1.C1(C)CC(=O)N1 c1(OC)ccc2[nH]c(=NC3CCN(C(=O)C(N)=O)CC3C)ccc2c1 Cn1c(C(N2CCN(CC(=O)NC3CC(=O)NC3=O)CC2)=O)ccc1C#N C1(C)(CNC(CC2N(CC)CCOC2)=O)CN(C(c2cnc(Cl)[nH]2)=O)C(C)(C)C1 C(=O)(C#CC1(C)CC1)NC1CCCN(C(C(N2CCN(C)CC2)C)=O)C1 c1(C(=O)NC2CC(C)(NC(C(C)N(C(C)=O)C)=O)C2)ccc(C2OCCO2)cc1 C12(NC(C3CCC(N=[N+]=[N-])C3)=O)CCCN(c3ncc(O)cn3)CC1C2 N1(C(C2N(C(c3c(COC)ccs3)=O)CC=CC2)=O)CC(C)OCC(C)(C)C1 c1(C(C)NC2CCCN(C(=O)COCCN(C)C)C2)ccc(O)c(F)c1.N(C)C Cc1ccc2[nH]c(C(N3CCC(NC(=O)CC4CCOC4)C(C)C3)=O)c(C)c2c1 Cc1nnc2n1CCN(Cc1cn(Cc3cnc4c(cnn4C)c3)nn1)C2 c1(C(N2CCC(CC(C)NC(C(CC)(C)F)=O)CC2)=O)cc(C)c(O)c(C)c1 C1(C(N(CC(=O)NC2CCCSCC2)C(C)C)=O)Cc2nccn2C1 CCCCC(CC(=O)N(CC(F)(F)Cl)C)NC(c1cc(C)nc(O)n1)=O C(=O)(C(CC(C)C(C)(C)C)N1CCOCC1C1CCCC1)NC(CCOC)C1CC1 n1(C(C)C)cc(C(=O)NC(C(=O)NCC(n2ccnn2)C)C2(C)CC2)cn1 c1(C(=O)NCCOCCOCCOCC)cc[n+]([O-])cc1.C1(CO)CN1 C1(CC(=O)NCC2(C)N(C(COCC)=O)CCC2)Cc2cc(F)ccc2O1 C1(C(=O)NCCCN(C(C2=C(C)CCC2)=O)CCO)CC2(C1)CC(C#N)C2 C(C)(C(=O)N1CCCC1CC(N1CCC(O)C1)=O)(C(C)C)OC O=C1CCC(C(=O)NCCCOCC(C)(C)NC(C2OCC3CCCC23)=O)=NN1 Cc1ccn(C(C)C(=O)NCC(c2ccccc2)NC(=O)C(O)C2CC2)n1 C1(NC(C2(C#N)CC2)=O)CN(C(c2cc(C(F)F)cc(F)c2)=O)C2(CCCC2)C1 C(c1cncc(F)c1)=CC(=O)NC1CC(C)(NC(C2C(CC)C2)=O)C1 C1(C)(C(=O)NCC(CC)NC(c2cnn(CCO)c2)=O)CC1(C)C C(N=c1ccnc(NC2CCCC2F)[nH]1)c1n(CC(C)C)ccn1 Cc1cnc2n1CCC(C(N1CCCC1(C)CNC(c1coc(Cl)n1)=O)=O)C2 C(=O)(C(C)(C)CCC#N)NCC1N(C(CN2C(=O)CC(C)(C)O2)=O)C2C(C1)C2 C(=O)(C1=CCCCCC1)NCC(F)(F)F.N12CCC3C(C3C1)NC(=O)CC2=O N1(C(C=CCCC=C(C)C)=O)CCCC2CN(C(=O)CNC(=O)C(C)(C)C)CC12 CC(C)C(C(=O)N1CCC1(C)C)OC(C(C)C)C1CC1c1ccccc1 C1(C(=O)Nc2cccc(C(=O)OCC)c2)CCC(C)CN1C(=O)NC1CC1(F)F C=CC(C)CC(=O)NCC1(COC)CN(C(C2(O)CC(C)(C)C2)=O)C1 c1(C(=O)NC2(C)CC(NC(CC(C)N(C)C)=O)C2)sc(Cl)cc1Cl N1(c2cc3cnc(C)n3cc2)CCn2ncc(S(C)(=O)=NC(=O)C3(Br)CC3)c2C1 N1(C(C(C)OCC)=O)C2CCC1CN(C(=O)C(C)CC(C)(C)C)C2 C#CCCC(O)C(=O)NCC1CCN(C(=O)C=Cc2ccccc2Br)C1 CC1(C)CC(CNC(c2ccc(=N)[nH]n2)=O)CN(C(c2ccn(CCF)n2)=O)C1 C1(CC)CN(C(=O)C=C(C)C(F)F)CCC1NC(=O)C(C)(C)C(=O)OC(C)(C)C C(=O)(C1=CCCOC1)N1CCCC(N(C(=O)COCc2ccnn2C)C)C1 C12(NC(c3scc(OC)c3OC)=O)CCC(CNC(C3CCC(=O)O3)=O)(C1)OC2 c1(C(=O)OC)cc(SC(c2sncc2C)c2nnnn2C)cc(F)c1 c1(NC(c2cccc(NCc3cnccn3)c2)=O)ccnc(CO)c1 N1(C(CSCC(=O)OC)=O)CCC(NC(c2ccco2)=O)CC1C1CC1 CCC(C)C(O)C(C)C(=O)NC(CC)(CC)CCNC(C1(C2CCCO2)CC1)=O C1(CNC(c2c(CC)cc[nH]2)=O)CN(C(c2ccc(SC)s2)=O)CCCO1 N1(C(C(=Cc2cccnc2)C)=O)CCCC(NC(=O)CO)CC1 C1(NC(CC(C)N(C)C)=O)CN(C(=O)CCOCc2ccccc2)CCC1C C1(C(=O)NCCOC2CN(C(c3cc(C(N)=O)no3)=O)C2)CC2CCC1O2 Cc1c(C=CC(=O)NCC2CC(NC(c3scc(Cl)c3Cl)=O)C2)cnn1C N1(CCCN2CC(C)C(O)CC2)CC2CCOC(=O)C2C1 C#CC1(O)CC(C(=O)N(CC(C)NC(=O)C(c2ccc(F)cc2)C)C)C1 C1(C(=O)NCc2cccnc2O)CC2CCC(C1)N2C(=O)COCC(F)F CN1CC(C(N2CCC(C(F)CNC(c3nnn(C)n3)=O)CC2)=O)CC1=O C(=O)(C1SCCc2ccccc21)NC1C2CN(C(c3c(C)[nH]nc3Br)=O)CC21 N1(CCNC(CCSC)(C)c2nnnn2C(C)C(=O)NC(N)=O)CCCCCC1 c1(CNC(C2(CC)CN(C(C)=O)C2)=O)ccc(NC(=O)OC(C)(C)C)cn1 c1(C(N(C(C)C(=O)NC(CNC(N)=O)(C)C)CC)=O)cc(C)c(F)cn1 c1(CNC(C(C)(N(C)C(=O)OC(C)(C)C)NC=O)=O)ccc2ccsc2c1 c1(C(=O)NC2CC(NC(c3cnn(C(C)C)c3N)=O)C2)c(Cl)ccc(F)c1C N1(C(CCN(C(=O)CC2CCC3CC23)CCO)=O)CCCC(O)(C2CC2)C1 C1(C(=O)NCC2(CC(=O)N(CC(F)F)CC#C)CC2)CCC(C)(O)CC1 N1(CCOC2CCCC2)CCC1C(N(C)CC)=O.C1(=O)CCOCCCN1 C(C(C)(C)CCN=c1[nH]c(N(C)CC2CCOCC2)nc2cc(C)ccc12)OC CCC(CCCC(=O)NCc1nc(C)ns1)NC(c1cc(C)on1)=O C(=O)(C1=C(C)OCCC1)N1CC(NC(c2cnc(CCCC)[nH]2)=O)C(C)(C)C1 CCCCCCC(C)C(=O)NCCC(O)CNC(=O)CC1CC(CC)C1 C12(C(N3C(CNC(Cc4cnc(C)[nH]4)=O)CN(C)CC3)=O)CC(C)(C1)OC2(C)C Cc1ccc(Br)c2cc(C(N3CCS(=O)(=O)CC3)=O)[nH]c12 N1(C(c2cn(C)nc2Cl)=O)CCOCC(CNC(C2(CO)COC2)=O)C1 c1(C(N(C2CCN(C(c3[nH]cc4c3CCCC4)=O)C2)C)=O)cnc2occc2c1 c1(C(N2CC(CC)N(C(c3ccnn3C)=O)CC2)=O)c(F)cc(OC)cc1F c1(C(N(C(C(=O)NC(CC)Cn2cncn2)C2CC2)C)=O)cc[nH]c1C c1(C(=O)NCC2CCC(NC(CC(C)C)=O)CC2)ccc(C(C)(C)C)c(Cl)c1 C1(OCO)CCN(N2CCC(Oc3cccc(Br)c3)CC2)C2(CCC2)C1 c1(OC(CSCCCC)=O)ccc(-c2cc(OC)on2)cc1 N(C1CCOc2cc(F)ccc21)C(C(=O)NC1(N2CCOCC2)CCCCC1)=O Cc1cc(S(N)(=O)=O)oc1C(=O)N(CCCCCNC(=O)CC1OCCC1C)C N1(C(C(C)NC(CC)(C)C)=O)CCC(O)(C(=O)N(CCC(=O)O)CCO)CC1 C1(CNC(CCC=C(C)C)=O)CCC2(CCC2)C1NC(=O)Cc1n[nH]c(C)n1 N1(C(c2cc(C)c(F)nc2)=O)CC(C)CN(C(=O)Cc2ccc(F)cc2)CC1C c1(CNC(CCC)c2ccco2)nc(Cl)nc(C(=O)OC)c1NC(=O)OC C(=O)(CCC(C)(F)F)N1C(C)CC(CC)C1.C(=O)CC(=O)NC C(CC(N)=O)(C(=O)NCCC1CCCOC1)NC(CCC1CCC(C)O1)=O C1(CCC)CCCN(C(C2(NC(c3cc(F)n(C)n3)=O)CCSC2)=O)C1 Cc1cnncc1C(=O)NC1C=CC(C(=O)NCCN(C)C2CC2)C1 c1(OC)c(C(=O)N(CCCN(C)C(c2cc(N)ccn2)=O)C)cccc1[N+](=O)[O-] Cc1cccc2ncc(CNCC3CCCC3c3cnn(C)c3)n12 C=C=CCCC(=O)NC(C1CCN(C(=O)Cc2ncccc2Br)C1)C C(C(C)(C)CNC(CCO)C1CC1)(c1nnnn1Cc1cccs1)NCCOC N1(C(C(C=C=C)C)=O)CC(C)(C)CCC1CNC(c1ncccc1CSC)=O N1(C(c2cccc(OC)n2)=O)CCC2CN(C(c3ccc(Cl)[nH]3)=O)CC2C1 CC(C)CCCCCC(=O)NCC1CN(C(c2cnnc(O)c2)=O)C2(CCC2)C1 C1(CNC(COCCC)=O)CC2(CO1)CN(C(=O)C=Cc1ccc(F)c(C)c1)C2 C(C(C)(C)C(C)(C)O)NC(C1(CSC)CN(C(=O)CN2C(=O)CCCC2=O)C1)=O C#CCCCC(=O)NCCCCCN(C)C(c1ccc(OCCOC)o1)=O CC#CCCCC(=O)N1CC(C(C(N2CC3CC(C)C3C2)=O)OC)C1 C1(NC(c2nc(CC)oc2)=O)CC(CO)N(C(=O)C(N2CCCC2)C2CC2)C1 N(C(=NCCSC)NCC(=O)Nc1cccc(Cl)c1)C1N(CCOC)CC1.C(CSC)N c1(C(=O)NC2C(NC(=O)CS(=O)(=O)NC3CCCC3)C2)cccc2nccnc12 CC1(C)CC(CO)CN(N2CCC(Oc3ccc(C#N)cc3Cl)CC2)C1 N1(C(C2(C(=O)NCC)CCCC2)=O)CCn2nc(COC)cc2C1 C(CCCC(=O)N1CC(C)(NC(=O)CCC(O)c2ccccc2)C1)OC C(=O)(C(O)C(C)c1ccccc1)N1CC(O)(CNC(CC2(C=C)CCC2)=O)C1 c1(C(=O)NC2CCN(C(C(CCCOC)C)=O)C2)nc(O)c2ccccc2c1C c1(NC(=O)NC(COCC)C)cccc(Nc2ccnn2C(C)CC)c1 N1(C(c2ccnc(C)n2)=O)CC(CC(=O)NC2CCOC(C)(C)C2)C2(CC2)C1 CCC(CC)CC(F)C(=O)NC1(C(=O)NCCC(O)C2CC2)CCSC1 N1(C(=O)Nc2ccc(Cl)c(C(=O)OC)c2C)CCC2(CCCC(CO)O2)C1 C1(C(=O)NCc2nnc(C)s2)CN(C(C)C(=O)NC(=O)NC2CC2)CCC1C CCCCCCC(C)CC(=O)N1CC2(CC2)CC1CNC(c1sc(CC)nc1C)=O C=CCC(CC)C(=O)NCC1(F)CCN(C(=O)Cc2csc(=N)[nH]2)C1 Cc1c(C(N2CCCC(CC(=O)NCC(C)(C)CN(C)C)CC2)=O)cccc1C#N C1(C(C)NC(C(=O)NCC)=O)CCCN(C(c2ccc(CN(C)C)[nH]2)=O)C1 N1(C(C2C(CC(C)C)C2)=O)CCN(C(C2CCC2)=O)C(c2cccc(F)c2)C1 c1(C(C)(C(F)(F)F)NC(Cc2c(C)cnn2C)=O)ccc(F)cc1F c1(C(N2CC3CCN(C(c4nn(C)c(O)c4)=O)C3C2)=O)ccc(Cl)c2occc12 Cc1nn(C)c2c(NC(C)C(C)C)nc(N3CCCCC(SC(F)F)C3)nc12 C(=O)(C1=CC2(CN(C(=O)C3CC3)C2)OC1)N(C(CC#C)C)CC C1(NC(CCN(CC)CC)=O)COC2(C1)CN(C(=O)C=Cc1c[nH]nc1C)C2 N1(C(C2C(=C)C2)=O)CC2(C)CN(C(c3ccc(OC)c(C)c3Br)=O)CC2(C)C1 CC1CCN(C(C2CCOCC2)=O)C(C)C1NC(c1cccc(N(C)C)c1)=O N1(C(c2c(C)n(C(C)C)nn2)=O)C2CCC1C(CNC(C1CCCC(O)C1)=O)C2 c1(C(=O)NC2CCCC(NC(C(C(=C)C)(C)C)=O)C2)ncnc2ccsc12 N1(C(CCC(CC)CC)=O)CC2CCCN(C(=O)C(O)CC(N)=O)C2C1 c1(CC(C(=O)NCC2OCCC(NC(C=CCCC)=O)C2)C)ccc(Cl)cc1Cl N1(C(c2ccc(OC)cc2)=O)CCC2(CC1)CC2C(=O)Nc1ccnc(Cl)c1Br N1(C(C(C(=O)OCC)OC)=O)CC2CCC(C(N3CCCC3CC)=O)(C2)C1 N1(C(c2cnn(CC)c2C)=O)CCN(C(=O)CC2CCC(O)C2)C(C)C1C c1(C(=O)NCC2CCCC2C(=O)NCC2CC23CC3(F)F)cc(F)cc(F)c1 C(=O)(CCCCCF)NC1CCN(C(C(CCC)OCC)=O)C1C N1(C(C(C)(C)OC)=O)CCC2(CCC2)C(CNC(=O)C(SC)SC)C1 CC1COCCN(C(=O)CC2CCN2C(c2ccc(F)c(O)c2)=O)C1 N1(C(COCC(=O)NC)=O)CCC(C(=O)NCc2ccn(C)c2)C1 c1(OCC)ccc2occ(C(=O)Nc3ccc(NC(=O)OC)c(C)c3)c2c1 C1(C(=O)NCc2scc(-c3ccc(C)cc3)n2)CC(F)(F)C12CC2 c1(C(C)OC)noc(CC(N2CCC(N(C(=O)CCc3nncn3C)C)C2)=O)n1 Cc1cc(C(=O)NCC(CC2CC2)C(N2CC3(CC3)CC2CO)=O)c[nH]c1=N C(c1cc[nH]n1)=CC(=O)NC1CC(C(N(C2(C)CCC2)CCC)=O)C1 c1(OC)cc(NC(C)CCCCNC(C2CCC=CCC2)=O)ncn1 C(=O)(CCCC(CC)NC(=O)CC(C)F)NCCC=C=C C#CCCCCCCc1nc(C2COCCN2Cc2nnnn2CC)no1 CC(C)(C(=O)N1CCOC(CNC(=O)Cc2cccnc2)C1)C(F)c1ccccc1 C1(CC(=O)NCCN(C(=O)CC2CCCC(C)O2)CC)CC(O)C1(C)C c1(C(=O)OC)ccc(C(F)(F)F)nc1.C1(F)C(=O)NC(C)(C)COCCN1.OCO C1(CC(N2CC(CC(C)NC(=O)CNC(c3ccoc3)=O)C2)=O)NC(=O)NC1=O C1(OC)CC(C(=O)Nc2ccc(C(F)(F)F)cc2O)CN(C(=O)C(C)=C(C)C)C1 C1(C(N(C(C)CNC(C2CCC(=O)N2)=O)CC)=O)CCCCC1N=[N+]=[N-] c1(NC(C2(CNCc3ccc(OC)c(O)c3)CC2)=O)cc2cccnn2n1 c1(C(=O)NC(CCC)CNC(c2cc(Cl)cs2)=O)cccc2nonc12 C1(OC)CC2(C1)CC2NC(=O)C(CC1CCCC1)NC(=O)C1=CCCO1 c1(C(=O)NC(c2ccc(O)cc2)CCO)ccc2nccnc2c1 CC(C)CC(C(=O)NOCC(O)CO)N(C(=O)C(C)c1ccsc1)C N1(C(c2cccc(C(F)(F)F)c2)C(=O)NC(CC)(C)C)CCC2(COC(C)C2)C1 N1(C(c2nc(OC)oc2)=O)CCN(C(=O)C=CSC)C(C)C1C N1(C(CC=C)=O)CCN(C(=O)Cc2ncc(C)s2)C(c2ccccc2Cl)C1 C1(CN(C(c2cc(COC)on2)C(=O)NCC)C)CCN(CC(F)F)CC1 c1(C(=O)NCC(CNC(c2ccc(CC)o2)=O)(C)C)cc2sc(C)cc2[nH]1 C#Cc1ccc(C2CC2C(=O)NC(C)CCNC(=O)CCCC2CCCC2)cc1 CC(C)(C)C1=NOC(C(N2CCCC2(C)CNC(=O)CC2C=CCC2)=O)C1 Cc1nc(C(N2CCOCC2CNC(=O)C(c2ccccc2)C)=O)nn1C C=CC(C)(CC)C(=O)NCCC1(CNC(=O)C(C)C(C)(F)F)CC1 n1(CC(N2CCC(C)(NC(C(C)OCCOC)=O)C2)=O)cnc([N+](=O)[O-])c1 Cc1c(CCNCC2CCC(C)CN2C(=O)C(F)(F)F)cccc1CO C(=O)(C1=CCN(C(c2c[nH]c3ccccc23)=O)CC1)NC1(C#C)CCCOC1 CC(C)C(C)C(=O)NCCC(O)C(=O)NCCC(O)C1CCC1 C(CCCC(CO)NC(=O)Cc1cc(Cl)no1)NC(=O)Cc1cnc[nH]1 Cc1ccc(NC(C2(C)CN(Cc3nc4ccccc4s3)C2)=O)c(F)c1F Cc1ccc(C(=O)NC2CCCN(C(=O)Cc3ccnn3C3CCC3)C2)c(F)c1F CN1CCN(C(=O)CC2CCSC2)C(C(=O)NCCCN=[N+]=[N-])C1 N1(C(C(C2CCC2)NC(C(C)n2ccnc2)=O)=O)CCC(C2(C)CC2)C1 C12(NC(c3c(C)cco3)=O)CCC(CC1n1cc(Cn3ccsc3=O)nn1)C2 C1(NC(C=CC=CCC)=O)CN(C(=O)C(c2ccccc2Cl)O)CCC1(C)C c1(C(=O)NCCN(C(=O)CNS(=O)(=O)C2CC2)CCC)ccc2ccccc2n1 Cc1ccccc1C(=O)N(C(C)CCNC(=O)C=Cc1nnn(C)n1)C Cc1ccc(NC(=O)C=CC(C)NC(c2ccnn2C(C)C)=O)cc1Cl N1(C(c2ccc(C)cn2)C(=O)NC(CC)C)CC2(C)CSCC2(C)C1 c1(C(=O)Oc2cccc(C=Cc3ccc(C(N)=O)o3)c2)cc(F)cc(F)c1 c1(CNC(C2CCN(C(c3ccc(C#C)nc3)=O)C2C)=O)c(C)nc(C)nc1C c1(C(=O)NCCCCn2cc(CCC3CCCC3)nn2)cn2c(n1)SCC2 Cc1ccc(N)c(C(=O)NC2CC(CNC(C3(C)CC3(C)C)=O)C2)c1F S(=O)(=O)(c1cccc(Cl)c1Cl)N.N#Cc1cnc(N(C2CC2)C=O)c(F)c1 N1(C(CN2CC(C)(C)C2)=O)CCN(C(c2[nH]nnc2C2CC2)=O)C2CS(=O)(=O)CC12 C1(N(C(C2CC2C(F)(F)F)=O)CC)CCCN(C(=O)CCCc2cccnc2)C1 C1(C(N2CCN(C(=O)Cn3cccn3)C(CF)C2)=O)COc2cc(Cl)ccc2C1 S(=O)(=O)(c1cccc(NC(=O)C(F)(F)F)c1)N1CCCC(N)C1 C(=O)(C1CCCn2cnnc21)NCCN(C(=O)CCN(S(C)(=O)=O)C)CCOC c1cc2c(cc1CN(C1CC1)CC1CC1)OCCC21CCCC1 CC1(C)CCN(C(=O)C2=CCSC2)C1CNC(C1CC2(CCCO2)C1)=O c1(CN=C(NCc2cnc(C)s2)NC(C)C)ccc2c(c1)CCCN2C C(CC(C)N=c1ccc2ncc[nH]c-2n1)NC(C(C)=C1CCCC1)=O C1(Cn2ccc(C(C(=O)NCCOC)N(C3CCCO3)CC)c2)CCCC2CC12 N1(CCC(=O)NC2CCC(CCNC(c3ccc(Cl)s3)=O)C2)CCCCCC1 N1(C(C)C)CCC(CC(N2CCC(C(C)NC(C3CCCCC3)=O)C2)=O)CC1 c1(CC)n[nH]c(=NCCN(C(=O)CCc2ccc(F)cc2Cl)C)s1.C(CN)S c1(C(N(C(CC)CC(=O)NCCC2(O)CCCC2)C)=O)nccc(C)c1N c1(OCC(=O)NCC2CCC(NC(C(CC)(F)F)=O)C2)ccc(Br)c(C)c1 C1(NC(c2c(CC)ocn2)=O)CN(C(=O)C=CC(C)C)C2(CCOC2)C1 c1(NC2CCC(SC)C2)nc2c(c(=NCCc3cc(C)n(C)n3)[nH]1)CCCC2 C(CC(C)(C)NC(C1CSCN1C(=O)C=C(C)C(C)(C)C)=O)OCC C1(NC(CC(C)(F)F)=O)CN(C(=O)CNC(N2CCCC2)=O)CC(F)(F)C1 N1(C(CNC(CC)=O)=O)CC2CC(O)C1C2NC(C1CC(O)(C(F)F)C1)=O c1(C(N(CCOCCN(C(C(CCCC)O)=O)C)C)=O)sc2nccnc2c1N C(CN=C(NCC(c1nc(C)no1)(F)F)NC1CCCC(C(N)=O)C1)OCC c1(C(=O)OC)ccc2nc(N3CC4CCC(C3)C4NC(C)=O)sc2c1 N1(C(Cc2n[nH]c(=NC)s2)=O)CCCC2CN(C(=O)C(C)NC(O)CO)CC12 C1(C(N2C(CCC#C)CCC2)=O)CN(C(=O)C(C)(C)N(C)C)CC(C)(C)C1 c1(C(=O)NCC(C(C)C)NC(=O)C#CC2CCCO2)cc2cc[nH]c(=O)c2s1 C1(NC(CC=CC)=O)COCC1NC(=O)C=CBr N1(C(=O)CCOC2CC2)CC2CCC1CN2C(C1(n2cncn2)CC1)=O c1(C(=O)NC(C2(O)CCN(C(C=NOC)=O)C2)C)nc(O)nc(O)c1F C1(N(C(N2C(C)(C(=O)O)CCC2)=O)CC2CCCC2)CC2(CC(OC(C)(C)C)C2)C1 C=CCCCCCCCC(=O)NC1CCC12CCN(C(=O)C=CS(C)=O)CC2 C1(C)(NC(c2c(OCC=C)cccc2)=O)CCN(C(=O)CC(C=C)CC)CC1 c1(NC(c2ccn(C)c2)=O)cccc(NC(C2CCNC(=O)C2)=O)c1 N1(C(C2(CNC(c3cc(O)ncn3)=O)CC(C)(C)C2)=O)CC2(CCC2O)C1 c1(C(=O)NC2CCC(C(=O)NC(C)C3CC3)C2)nc(C)c(C)s1 C1(C(=O)NCCOCCN(C(=O)CO)C)CCCC2CCCN12 C=C(C)CCCC(=O)NCC1CCCCC1NC(=O)Cc1c(F)cccc1F C1(C2CC2)(NC(C(C)Oc2cccnc2)=O)CCN(C(=O)C2=CCCOCC2)C1 c1(C(N2CCOCC(NC(C3(COC)CC3)=O)C2)=O)c(F)ccc(Cl)c1F C(=O)(C(C(C)(C)C)C1CC1)N1CCC(N(C(CC(=O)NCC#C)=O)CCC)C1 C1(CNC(N(c2ncccc2-c2nccs2)CCC)=O)CCN(C)C1CC N(C(=NCCS(=O)(=O)C(C)C)NCCNc1c(OC)cccc1F)CC Cc1ccc(C(N2CCC(NC(=O)C=CC(C)C)C(CO)C2)=O)c(N)n1 c1(OCC)cccc2[nH]cc(CC(=O)N(C)CCN(c3ncc(C)cn3)C)c12 CCC1=NOC(CC(N2CCC(C(F)F)(CNC(=O)CCOC)C2)=O)C1 Cc1ccc2cc(CNC(=O)C(=O)NCc3ccc(C(F)(F)F)cc3)ccc2n1 CC1CCC(C(=O)NCC2C=CCCC2)N(C(C2CC3CCCC3C2)=O)C1 CC1OC2(CO)CC1(NC(=O)C(C)N(C(=O)COCc1ccccc1)C)C2 N1(C(c2ccc(C)s2)=O)CCCC(N(CCO)C(C2(C)COC2)=O)CC1 C(=O)(CCCC(=O)N1CC2C(CNC(c3ccncc3Br)=O)C2C1)NCCC C(C(C)(CC(=O)Nc1cccnc1-c1ccncc1)C(F)(F)F)N(C)C C1(CNC(CC(C)N(C(c2c(OC)n[nH]c2)=O)C)=O)CC2(C1)CC(O)C2 c1(C(=O)NCCC(C)NC(C2CCCS2)=O)ccc(OC(F)(F)F)nc1 C(CS(=O)(=O)c1ccc(C)cc1)N1CC(CCC)OCC1 CC1N(C)CCC1(c1nnnn1C1(C)CC1)NCc1ncoc1-c1cccs1 Cc1nc(O)c2cc(C(N3CCC(O)(c4ccc(Br)cc4)CC3)=O)ccc2n1 C1(N2C(C(N)=O)CCC2)CCN(CC(C)CC2CC2)CC1 c1(NC(N)=O)ccc(Cl)c(C(N2CCC(NC(=O)C=CC3CCC3)CC2)=O)c1 Cc1cc(CC(N2CC(N3CCN(C(C4CCCSC4)=O)CC3)C2)=O)ccc1F C1(NC(CC2N(C)C(=O)CC2)=O)CCC(O)CN(C(=O)Cn2cnccc2=O)C1 N1(C(Cc2scc(CC)n2)=O)CCCC1(C)CNC(c1c[nH]nc1F)=O c1(C(C)C)cnccc1CC(=O)NCC(C)(CO)NC(=O)C(=Cc1c[nH]cn1)F N1(C(C(CCC)NC(N)=O)=O)Cc2ccccc2C(CNC(C2CC2C)=O)C1 C1(NC(c2c(OC)nsc2)=O)CCCCN(C(c2ccc(F)cc2Br)=O)C1 c1(CCC(=O)NC(C)CN(C)Cc2cccc(F)c2)ccc2ocnc2c1 CCC(C)(C)C(O)C(=O)N(CCCNC(C1CCCSC1C)=O)C1CC1 O1NC(=O)CC(COC)NC(=O)C1.C1(C(C2CCCO2)(C)C)CC(=O)C12CCC2 N1(C(C(=O)Nc2ccc(C)c(Cl)c2)=O)CC2CC1CCN2C(C1CC12CCC2)=O C(=O)(C1Cc2ccccc21)N1C(C)CN(C(C2CC2CF)=O)CC1 C1(C)(C(=O)NCC(CNC(c2ccc(SCC)cc2)=O)(C)C)CCC(C)=C(C)C1 N1(C(c2cn(CC)nc2)=O)CC2CCCC(NC(C3(Cl)CC3)=O)C2C1 c1(C(=O)NC2CC(CNC(CCC=C)=O)C2(C)C)ccc(C)c(C)c1O c1(OCC)cccc(CNC(=O)NOc2ccc(I)cc2)n1 C1(NC(c2ccc(CO)cc2)=O)CN(C(c2ccncc2)=O)C2CC12 C(C(=O)NC1CC(CC(=O)NCCC23CC(CCO2)C3)C1)(C(C)(C)C)OC N1(Cc2cccc(C)c2)CCNCC2CCCCC12 CN1CCN(CC(=O)N(C2CCN(C(=O)C=Cc3ncco3)C2)C)CC1=O C1(C(=O)NCCNC(c2cc(COC)[nH]n2)=O)CC(=O)NC(=O)C1 CC1CCN(C(=O)CCC(F)(F)F)CC1NC(C1CCC2CC2CC1)=O CC1CN(C(=O)CC2CC2(Cl)Cl)CC1NC(C1CCCN(c2cnccn2)C1)=O C(=O)(CS(=O)(=O)C1CC1)NCC(=O)N(C1(C#C)CC1)C N1(C(C2(C)CNC(=O)C2)=O)C2CCC1C(F)C(NC(c1cc(CCO)on1)=O)C2 CC1CN(c2cc(Cl)nc(CO)n2)CCC1CNC(=O)COC1CCCCC1C CC1(NC(=O)C=Cc2ccc(O)cc2)CCCN(c2ncc(Br)c(O)n2)C1 C1(C(=O)NCC(CNC(c2c(C(C)C)onc2)=O)F)CCC(F)(F)CO1 C1(C(=O)NCC(CC)N(C)C(C)=O)CCN(C(=O)C2CC2)C1(C)C N1(C(c2ccn(CC)c2C)=O)CC=C(CC(=O)N2CCCSCC2C)CC1 c1(CNC(=O)C=CC(N2CCC23CN(CC)C3)=O)ccc2cnn(C)c2c1 Cc1cccc(Cl)c1CC(=O)NC1CC(NC(=O)C(C)CC2CC2)C(O)C1 c1(OC)ccc2c(c1)cc(C(C(=O)NCC(C)C)NC(c1ccccc1)C)n2C N#Cc1cccc(C(N2CCC(F)(F)C(NS(=O)(=O)c3cccnc3)C2)=O)c1Cl c1(C(N2CCC(C)(CNC(=O)CC3CCC(=O)N3)C2)=O)ncc(Br)cc1N c1(-c2cc(C(=O)NCCC3CN(C(C(C)=C4CC4)=O)C3)on2)ccc(F)cc1 C1(NCC(n2cc(Cl)cn2)C)(Cc2ccccc2)COc2ccccc2C1 c1(NC(N(C)Cc2cccnc2)=O)ccc([Si](C)(C)C)cc1 C1(C(=O)OC)CC(=O)N(C)C1C(=O)NC1CN(C(=O)CNC(N)=O)C(C)(C)C1 CCC(C)CC(=O)N1CCN(C(C2C=CCS2)=O)CC1 C(=O)(CCCCC(F)(F)F)N1CCC2(NC(CN3CCC(OC)C3)=O)C(CC1)C2 c1(C(N2CCCC(C)(F)C2)C(=O)NC(C(=O)OC)C)cnc2ccccc2c1 c1(CCNC(c2oc(Br)nc2C(F)F)=O)cc(F)ccc1F N1(C(C(C)SC(F)(F)F)=O)CCCN(C(c2cnc(-c3cccs3)o2)=O)CC1C CC1(C)CCN(C(c2ccc(CO)o2)=O)CC1C(N1CCC2(CO)CCCC12)=O C1(C(=O)NCCCSCC)CCC(C2CC2)N1C(=O)C(C1CCCCC1)C C1(CNC(Cc2nc(C)oc2)=O)CCCN(C(=O)CCCn2cccn2)C1 N1(C(CCc2c(C)nn(C)c2)=O)CC2=C(C1)CN(C(C1CC(OC(C)C)C1)=O)C2 C1(C(=O)NCC(CC)NC(=O)CSc2nnc(S)s2)CCCCC12CCC2 C1(NC(C2CC(C)(C)OC2)=O)CN(C(c2cc(Cl)cc(N)c2F)=O)C2(CCC2)C1 C1(C(N2CC3CC3C2)=O)CC12CCN(S(=O)(=O)CCn1cnc3ccccc13)CC2 N1(C(CN(C(C)=O)C)=O)CCN(C(c2sccc2Oc2ccn(C)n2)=O)CC1 CC1(C)CCC(C)(C(=O)NCC(C2CC2)NC(=O)CC(O)C(Cl)(Cl)Cl)CC1 CC1CCOCC1C(N1CCC2CC12C(N1CC2CC2(CO)C1)=O)=O C1(C(N2C(CC(=O)N(C3CCCC3C#N)C)CCC2)=O)CC2(C1)CC(O)C2 N1(C(c2nccc(C)n2)=O)CCC2(CCN(C(c3cc(C)c(C)n3C)=O)CC2)C1 C(=O)(CCCCC(=O)OC)N1CC(NC(CCCOCC)=O)C(F)C1 Cc1nn(C)c(C)c1CCC(=O)NCC1C2CC1N(Cc1ncco1)C2 c1(C(=O)OC)c[nH]c(NC(C)CC(C)NC(=O)C(n2nnnc2C(C)(C)C)C)c1 C1(S(=O)(=O)N(C2CC3CC2CN3C(=O)CO)C(=O)OC(C)(C)C)(CC=C)CCC1 Cc1cn2cc(CC(=O)NC3CCC3CNC(=O)Cc3ccc(F)cc3)nc2s1 CC1(C(N2CCCC(CF)C2)=O)CCN(C(=O)C(O)CC2CCCC2)CC1 N1(C(=O)Cn2nnc(=O)[nH]2)CC2CCC(C1)N2C(c1cn[nH]c1)=O N1(C(c2n(C)cc(Br)c2)=O)CC2CC(O)C1C2NC(=O)CCC(C)(C)C N1(CC2C(C#C)C2)CCC(OCC)C12CC2 C1(NC(CN(C)C2CC2)=O)CCC(C(=O)NC2(CCO)CCOC2)CC1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CC(F)CC(C(=O)Nc2ccc(CC)cn2)C1 N#Cc1ccc(Br)c(C(N2CCCC2C(=O)Nc2cnn(CCO)c2)=O)c1 CCC(C)(F)C(=O)NCCC1CC(NC(c2cc(C3CCC3)[nH]n2)=O)C1 N1(C(C(CC)N(CC)CC)=O)CC2(C(N3CCCN(C)C(=O)C3)=O)CCC1CC2 N1(C(Cc2nc(CC)sc2)=O)CCC2(NC(c3cc(C4(C)CC4)on3)=O)CC2C1 C(=O)(C(CC(C)C)C(C)C)N1C2CC(CNC(C3(OCC)CCC3)=O)C1CC2 N1(C(Cc2nn(C)c(=O)n2C)=O)CC2CCC1CN2C(C12CSCC1C2)=O c1(C(=O)OC)ccc(C(=O)NC2(C(C)C)CCC2)cc1.C12CC1CNC2=O c1(NC(C2C=CC(NS(CCCC)(=O)=O)C2)=O)nc2cccc(Cl)c2s1 N1(C(CNC(CC(=O)OC)=O)=O)CCC(N(CCCO)C)CC1.C1CCO1 c1(COc2c(NC(CN(C3CC3)CC)=O)cccn2)ccc2c(c1)OCO2 c1(C(=O)NCC2C(NC(c3cc(C)n(C)c3C)=O)CCC2)cscc1S(C)(=O)=O N1(C(CNC(CC)=O)=O)C2CCCC1CN(C(c1ccccc1S(N)(=O)=O)=O)C2 c1(C(N2CC(CN(C(C3OCC(C)C3)=O)C)C2)=O)ccc(C(F)F)cc1 c1(NC(c2cccc(SC)c2)C)[nH]c(=NC2CCSCC2)nc2scnc12 N1(C(CCOCC#C)=O)CCN(C(CNC(C2(C(C)C)CC2)=O)C(F)F)CC1 C1(NC(C(COC)(C)OC)=O)CCCCN(C(C2(CCO)CC2)=O)C1 c1(C(N2CCC(O)(CNC(C(CC)(F)F)=O)CC2)=O)ccc2c(c1)OC(C)(C)C2 c1(CC)cc(C)ccc1C(=O)NCC1CC1CNC(=O)CN1CCCNS1(=O)=O N1(C(CCOC)=O)CCOCC1(C)C.c12cncc(c1)C(=O)N2 C(CCC(=O)N1CCCC1CCN(CCOC)CC)NCCC S(=O)(=O)(c1cnn2cc(Br)cnc12)NC(C(C)c1ncco1)=O C(=O)(C1=CCCCC1)NC(C(=O)N(CCOCC=C)C)CC1CC1 Cc1cccn2cc(C(N3CCN(C(c4nonc4N)=O)CCC3C)=O)nc12 Cc1cc(C(N2CC(OCCNC(C3CC4CCCC4C3)=O)C2)=O)ncc1Br N1(C(C(CN(C)C)N(C)C)=O)CCC(C(=O)N(CC(C)(C)C)C)CC1(C)C N1(C(CCS(C)=O)=O)CCOC2(C1)CN(C(c1ccc(N)cc1Cl)=O)C2 C=CCCCC(=O)NCCCC(C)(C)NC(=O)CCC=CC C1(N(C(COCC=C)=O)C)CCCN(C(=O)C(c2cccc(O)c2)C)C1 N1(C(C(C2N(C(CC(C=C)CC)=O)CCC2)(C)C)=O)CCOCC(C)(C)C1 C1(C(C)=O)CCN(CC(N2CC3CC3(NC(c3cc(C)c[nH]3)=O)C2)=O)CC1 c1(C(=O)NCC(C)(C2CCC2)NC(=O)Cc2ccccc2)coc2c1CSC2 C(CCOC)(C(C)C)NC(C(C1CC1)NC(CCCOC)=O)=O C(=O)(C(C)CCC(=O)OC)NCc1c(CNC(CCCC#CC)=O)cccc1 c1(C(=O)NCCC(C)CCNC(C2CC(=C3CC3)C2)=O)nnc(O)nc1O Cc1cc(OCC(O)CNc2cccc(N3CCN(C)C(C)C3)n2)cc(C)c1 N1(C(c2cnc(N(C)C)o2)=O)CC2(CCC(C(N3CCCCC3C#N)=O)O2)C1 C1(CNC(c2cn(CC=C)nc2)=O)CCC12CCN(C(=O)CNC(N)=O)CC2 CCCCCC(CCCCC)C(=O)N1CC2CC(O)C1C2NC(=O)CC(=O)NC C(=O)(CCCC(=O)NC(C)(C)CCCNC(=O)C(C)(CC)CO)NCC c1(-c2nc(-c3c(C)occ3)nn2C(C)C(F)(F)F)cc(S(N)(=O)=O)c[nH]1 C=CC1(NC(C2CC(O)CN2C(=O)C(C)C#N)=O)CCOCC1 N1(C(C(C)OC)=O)CC2(CCC(NC(=O)C(C)Cc3ccc(F)cc3)CC2)C1 N1(C(C2(CCC=C)CN(C(C3CC=CCC3C)=O)C2)=O)CCC(CC)(CO)C1 c1(C(N2C(CNC(c3c[nH]c(=O)cn3)=O)CC(F)C2)=O)cc2c(cn1)OCCO2 c1(C(=O)NC2C(C3CCN(C(CC(=C)C)=O)CC3)C2)ccc(OC)nc1Cl c1(C(N(CCN(C(c2c(CC)[nH]nc2Cl)=O)C)C)=O)ccc(OC)c(Cl)c1OC C1(NC(c2c(C)cccn2)=O)CC2CC(C1)N(C(=O)CCCC(C)(C)C)C2 N1(C(C=COCC)=O)CCN(C(C2CC3CCC3C2)=O)CC1CC Cc1cc(N)c(C)nc1C(=O)NC1(CNC(=O)Cc2ncoc2C)CC1 c1(CNC(=NC)NC2CC2C(C)(F)F)ccccc1F C1(C(=O)NCC(CC=C)NC(=O)C(F)(F)c2cccnc2)CCN(CC)C1(C)C C1(C(=O)NC2(CF)CCN(C(=O)Cc3c[nH]nc3O)C2)Cc2cscc2C1 Cc1ccc(=NC(=O)C2(N)CC(c3ccccc3)C2)[nH]n1 C1(C(=O)NCCc2nc(CC)[nH]n2)CCN(C(c2cnccn2)=O)C1CC c1(C(N2CCN(C(C3CC(CC)C3)=O)CC2C(C)C)=O)ccc2oc(O)nc2n1 C1(C(=O)NC23C(CN(C(C4(C(C)C)CC4)=O)C2)C3)CC2(C1)CC1(CCC1)C2 C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(c2cc(N)ccn2)=O)C2CCCCC12 C(C(=O)NCC(C)CC(F)(F)F)(C(C)(C)C)NC(C(C)OCCOC)=O.OC N1(C(COC(CC)C)=O)CCC(CNC(=O)CCC(F)F)C(C)C1 C1(=O)C(OC)CN1.C(=O)(CCCOC(C)C)NCCCOCCCC C1(CC(=O)NCc2c(C(=O)NCC(C)(C)N3CCCC3)[nH]cc2)CCC(=O)CC1 Cc1ccc(F)c(C(=O)NC2CC(C)(NC(C3CC34CCCOC4)=O)C2)c1F c1(OC)cc(C(=O)N(CCNC(=O)C=CC2CCCCC2)CC2CC2)ccc1C c1(OC)ccc(Cl)c(CC(N2CCC(C(N3CC4CCCC4C3)=O)C2)=O)c1 C1(NC(=O)C=CC(=O)NC2CC2)C=CCCN1C(C1CCC(O)CC1)=O Cc1cc(CCC(N2CCC(N(C)C(C3CC(=O)C3)=O)C2)=O)ccc1Br C1(CNC(CCC=CC)=O)(CNC(C2CC2C2CC2)=O)CC12CCC2 C1(NC(CCCC=C)=O)CCC12CCN(C(C1CCc3nnc(C)n3C1)=O)CC2 C(c1ccc2ccccc2c1)=CC(N1CC(CNC(CC)=O)CC1(C)C)=O N1(C(c2ccc(CC)s2)=O)CCCC(C(C)(O)CNC(=O)CN(C)CCO)C1 Cc1ccc(F)cc1C(=O)NCCC1CN(C(=O)C(C)CF)CCCO1 C1(OC)CC(C(=O)NCC(Cc2ccccc2)NC(C2(C)CC2(F)F)=O)CC1OC C1(CCC)CN(C(c2nocc2C)=O)CC1NC(C1CCC1)=O N1(C(c2ncccc2Cl)C(=O)NC(CC)C)CC2CCC1(CO)C2 Cc1cc(C(=O)NC(C)C(C)(C)NC(=O)CC(F)F)c2cc(F)ccc2n1 c1(C(=O)NC2(CCC(=O)NC(c3cccnc3)C)CCCC2)cc(F)cc(F)c1 C1(C(=O)Nc2nc(CN3CCOCC3)cs2)C2C=CC(O2)C1CO c1(C(N(C)CC2CCN(C(CCCC)=O)CC2)=O)cc(C(=O)OC)ccc1F c1(C(=O)NCC2(OCC)CN(C(CCCCC)=O)C2)ccc2ncnn2n1 C(CCC(C)CC(=O)OC(C1CSC1)=O)=C(C)C c1(C(=O)NCC2N(C(C3(C(C)(C)C)CCCC3)=O)CCC2)ccc(Cl)cc1N C1(C(C)NC(=O)C(C)n2cccn2)CN(C(=O)CN2CCS(=O)CC2)CCO1 C#Cc1ccc(F)c(C(=O)NCCC2CCC(NC(C3CC(CCO)C3)=O)C2)c1 N1(C(c2cccc(OC)n2)=O)CC(CNC(=O)C2=NOC(C)C2)C2(CC2)C1 CCC(CC(=O)NC(c1ccc(F)cc1)CNC(c1cncs1)=O)CC(C)C CC(C(F)(F)C(F)(F)F)=CC(=O)N(CC(O)CNC(=O)Cc1c(C)noc1Cl)C C1(C(=O)NCC(C(=O)NCC(N(OCC)C)=O)(C)C)CCCC1C1CC1 c1(CC2(C(=O)Oc3c(C)nsc3)CCC2)ccc(Cl)cc1 c1(C(N2CCC(OC)(CNC(=O)C=C3CCCC3)CC2)=O)nc2c(s1)COCC2 Cc1ccc(OCC(N2CC(CN(C(=O)C(c3ccccn3)O)C)C2)=O)cc1C C(=O)(C(F)(F)CC(=O)N1CC2CCC(NC(c3cncc(Cl)c3)=O)(C2)C1)OC N1(C(C(CSC)OC)=O)CC(CNC(c2cnc3n2CCC3)=O)CC(C)(C)C1 C(=O)(C1CCc2cccnc21)NC(C)CN(C)C(c1cc(Cl)ncc1N)=O C(CC(=O)NC1CCC(NC(=O)C(C2CCCO2)C2CC2)CC1)(C(C)C)OCC c1(C(N)=O)ccc(CCC(N2CCC(n3cc(-c4ccns4)nn3)C2)=O)s1 C1(O)(C(=O)NCC2C(C(N(C3CCCNC3=O)C)=O)CCC2)CCCCC1 N1(C(C(C2CCCCC2)NC(=O)C=CC(F)F)=O)CCCC(O)CC1 c1(OC)nc(C(=O)NC(CNC(C2(F)CCCOC2)=O)C(C)C)sc1C c1(OCC)cc(NC(C2CC2C(=O)Nc2cc(Br)cnc2Br)=O)c(Br)cc1F CC(C)C(F)(F)CC(=O)NC(C1CCN(C(C2CC3(C2)CC(C)(C)C3)=O)C1)C CC1(C(=O)NC2CN(C(c3ccc(S(N)(=O)=O)nc3)=O)C2)CCOC12CC2(F)F C1(NC(c2cc(C3CC3)[nH]n2)=O)CCCC(CO)C1.N12CC(F)(C1)C2=O C1(F)(C(=O)NC2CCC(NC(CCNC(C(C)(C)C)=O)=O)CC2)CCCCCC1 C1(CNC(N(C2CCN(CC(F)(F)F)CC2)C)=O)CC2(C1)CC21CCC1 C1(C(=O)NC2(C(N(OC)C)=O)CC2)C2CN(C(=O)CC3C=NN(C)C3=O)CC12 Cc1cccc(N)c1C(N1CCC(C)(CNC(C2CC2C2CCC2)=O)CC1)=O C1(C)(CNC(CC(C)n2ccnc2)=O)COCCN(C(c2cnc(O)n2C)=O)C1 CCC(C)CCC(=O)NCCC1(NC(=O)CNc2cccc(C#N)c2)CCC1 c1(C(N(CCCNC(c2c(CN(C)C)cco2)=O)C)=O)ccc(Cl)cc1[N+](=O)[O-] n1(CC(=O)N(CC(CNC(C=C(C)C2CC2)=O)C)C)nc(C)cc1C c1(C(=O)NC2CCC(NC(c3ccc(C#N)cn3)=O)CC2)coc2ccccc12 CC(C)CC(C)(C)CNC(C1CCCCCN1C(C1CCS(=O)CC1)=O)=O c1(C(N2CCN(C(c3cc(SC)c(C)o3)=O)C(CO)C2)=O)sc2nccn2c1C N1(C(c2c(C)nn[nH]2)=O)CC2CCCC(NC(=O)CC3(C(F)F)CC3)C2C1 C1(CNC(CSCC)=O)CCN1C(=O)CN(CC(C)(C)C)C C1(N(C(=O)C(=CC2CCCCC2)F)CC)CCCN(C(=O)CCC2CC(C)C2)C1 C1(NC(C2N(C(N)=O)CCC2)=O)CC2(C1)CN(C(C1(Cl)CC13CCC3)=O)C2 C(=O)(C(C)C(C)(C)C)N1CCN(C(Cn2c(C)ccn2)=O)CC1 C(=O)(C(F)C(F)(F)F)N1C(CC)C(C(=O)NCC2CCC3(CC3)C2)CC1 c1(C(=O)NC2(C)CCN(C(C3CC4(C3)CS(=O)(=O)C4)=O)C2)cc2nc[nH]c2cn1 c1(CC(N2CCN(C(c3nc(C)[nH]n3)=O)CC2)=O)c[nH]c2cccnc12 Cc1cc(=O)c(C(N2CCC3(CCCN3C(=O)C3CC3)C2)=O)cnc1C C1(C(N2CCC(O)(CNC(c3cnc(S)nc3)=O)C2)=O)SC2C=CC1CC2 C1(C(N2CCC(C(=O)NC)C2)=O)CN(C(c2cccnc2C)=O)CCO1 N1(C(c2c(C)cc(OC)nc2)=O)CC(C)CN(C(=O)CCC(F)(F)F)CC1C Cc1ccc(C(=O)NCC2CCC2NC(=O)CC(C)P(C)(C)=O)c2c1CCCN2 CC(C)C(C(=O)NCCCN1CCOCC1)C(C)NC(=O)C=Cc1cscn1 C(=O)(C1=COCCO1)N1CC(CCC)C(NC(=O)CCc2cnoc2)C1 C1(C)(COC)C=CCN1C(C1C=CC(NC(C2CC(N=[N+]=[N-])C2)=O)C1)=O c1(C(N(CC(C)(C)CNC(=O)C=CC2CCC2)C)=O)ccn2nnnc2c1 N(C1CCCn2nccc21)C(C#CC(CNC(C1C(=C)C1)=O)(C)C)=O C1(CCN(C)C(C2CCN(CC)C2)=O)CCN(C(c2ccc(OC)s2)=O)CC1 N1(C(CCCOC)=O)CC2(CCN(C(c3sc(NC4CC4)nc3C)=O)C2)C1 CC(C)C(C#N)C(=O)NC(C)CC(C)NC(c1ccccc1N(C)C)=O C#CCC(C)(C(=O)N1CCCC(OCC)C1)NC(=O)C=CC=CC C1(CNC(C(CCSC)(C)C)=O)CCC2(CCOCC2)CO1.C12CCCN1C2=O N1(CC(C)Cc2ccccc2)CCCCC(Cn2cc(C3CCC=CO3)nn2)C1 c1(CC)nocc1C(C(=O)NCC(F)F)N(CC)Cc1cnn(C)c1 C12(C(=O)NC(CC(N3CC4C(CC)(C4)C3)=O)(C)C)CCC(CC1F)C2 Cc1ccc(CN2CCCCC2C(=O)NC2CCOCC2F)cc1 c1(SC)ncc(C(N2CC(C)(NC(C34CC(C)(C3)C4)=O)C2)=O)s1 N1(C(C)=O)CCCCC1C(=O)NCCC1CCN(C(=O)Cc2nc(=N)s[nH]2)C1 C1(C(=O)NCC2(OCC)CN(C)C2)CC2CN(C(c3c[nH]nc3C)=O)CC2C1 C1(CNC(C(C)(C)C)=O)CCN(C(=O)CC23CCC(C)(C2)OC3)C1(C)C C12(CNC(c3nc(COC)oc3)=O)CCCC(CN1C(=O)C(C)=C1CCC1)C2 C12(C(=O)NCCN(C(Cc3nc(C)[nH]n3)=O)C)OCCCC1C2(F)F C1(C(=O)NC2CC(NC(c3c(C(C)C)noc3)=O)C2)CC(S(C)(=O)=O)C1 c1(C(N2C(NCc3cn(CC(C)O)nn3)CCCC2)=O)ccc2nsnc2c1 c1(C(=O)NC2(CO)CN(C(CCCC(=O)OCC)=O)C2)ccc2c(C)[nH]nc2c1 N1(C(c2nc(C)oc2C)=O)CCCC(NC(=O)C(c2ccc(F)cc2)(F)F)CC1 C1(CNC(CCN(c2ccccc2)C)=O)CCN(C(=O)CC2(C)CC2)CC1O CCCCC(C)(F)C(=O)N1CCOCC(C(=O)N(C2CCNC2=O)C)C1 c1(CCNC(N(C(C2CCCCC2)C)C)=O)ccc(C(N)=O)cc1 C1(CC(=O)NC(C(=O)OCC)CN(C)Cc2ccccc2)CCN(C)S1(=O)=O C1(C(=O)NCCCN(C(Cn2c(C)ccn2)=O)C(C)C)CN(C)CC1C C(C(=O)N(C(C)CNC(c1cccc(N2CCCNC2=O)c1)=O)C)(C(C)C)SC C#CCC(CC(=O)N1CC(O)(COC)C1)NC(C1CC1C(C)(C)C)=O Cn1cc2c(n1)CC(C(N1CC=C(CNC(C3COCCN3C)=O)CC1)=O)CC2 C1(C)(CNC(Cc2cnc(C)s2)=O)CN(C(c2c(F)cccc2F)C)CCO1 c1(CNC(CCCc2cn(-c3ccc(C)cn3)nn2)=O)c(C)nn2cccnc12 C1(CCNC(c2nc(Br)c[nH]2)=O)COCCN1C(C1CCCCS1)=O C1(C(=O)NC2CC(NC(C(C)CC3CCCC3)=O)C2)CN(C)CC1C(F)(F)F N1(c2n(CC(=C)C)c(-c3cnn(C)c3)nn2)CC(CO)C(C)(C(F)(F)F)C1 c1(CC)cccc(F)c1C(=O)NCC12CC(NC(=O)COC3CC=CC3)(C1)C2 N1(C(C(=O)OCC)=O)CCN(C(C2OCCC2OC)=O)CC(C)C1 Cc1ncc(C(=O)NCC2CC(NC(c3ccn(C)n3)=O)C2)[nH]1 N1(C(c2cccc(C(C)C)c2)=O)CC2(NC(=O)C3CC3)CCC1CC2 C(C(CC1CC1)C(=O)N(c1ccc(F)cc1)C(C)C)NC(C(N1CC(C)C1)C)=O Cc1nn(C)c(C)c1C(=O)NC1(C#N)CCN(C(c2cc(Br)ccn2)=O)C1 Cc1ccncc1-n1cc(CNC(=O)C(=O)NCC(O)C(C)(C)C)nn1 Cc1cc(NC(C2CC(C)CN2C(c2ncccc2N)=O)=O)c(C)c(C)c1 n1(CC)ncnc1C(N1CC(C(N)=O)(CNC(=O)C(c2ccccc2)F)C1)=O Cc1ccc2c(=NCC(C(C)C)OCCO)[nH]c(=NCCO)[nH]c2c1 C1(NC(C(C2(O)CCC2)NC(C=CCC)=O)=O)CCC(=O)NC1(C)C CN1Cc2cc(S(=O)(=O)NCC3Cc4cc(Br)ccc4O3)ccc2OC1=O C1(C(=O)NCC(C)(C(C)C)NC(CCC(=C)Cl)=O)CCC(C)(C)OC1 N1(C(C)=O)CCCCC1C(=O)NC(CO)C(C)NC(=O)Cc1cncc(O)c1 CC12CCC(C(N3CCCN(C(=O)CN4CCCCC4)C(CO)C3)=O)(CC1)CC2 Cc1cccc(C(N2CC3(CC(NC(C4CCS4(=O)=O)=O)CO3)C2)=O)c1[N+](=O)[O-] Cc1ccc(CC(=O)NC2CCCCC2C(=O)Nc2cnc(C)s2)cc1 CCC(C)(COC)C(=O)NCc1csc(CNC(=O)CC(C)(C)C)n1 c1(C(N2C(CCNC(C=CSC)=O)CCCC2)=O)cc(F)cc2ccoc12 C1(CC(=O)N(CCCC#C)C)CN(C(C2CC=CCC2)=O)CC1C N1(C(COc2cccc(C#N)c2)=O)CCN(C(c2ccco2)=O)C2CCC12 c1(-n2ncc(C(=O)NCC(CNC(C3CCCO3)=O)OC)c2)cccc(C)c1 n1(C(C)C)ccnc1C(N1CCC1CNC(C1CCCC1C)=O)=O S(=O)(=O)(c1ccc(Cl)cn1)NCC1N(S(CCC(=O)OC)(=O)=O)CCC1 N1(C(C(COCC)C)=O)CC(C)N(C(=O)CC2CC(CC)C2)CC1C C1(NC(CCCc2ccc(C)s2)=O)CCCN(C(=O)CCC2CCCN2C)C1 C1(NC(c2c(C(=O)OC)cco2)=O)CCOC(C(=O)NC(C2CCCC2)COC)C1 C1(CCC(=O)N(CCC(=O)N(C(CCC)C)CC)C2CC2)CCC(=O)C1 c1(C(N2CC(CC(C)NC(C=CSC)=O)C2)=O)ccc(C(F)(F)F)cn1 N1(C(c2nn(CC)nc2C)=O)CCN(C)CC1C(=O)NC(C)CSC(F)F c1(OC(C2(CC)CCO2)=O)nnc2c(c1C#N)CCCC2.C1CCC(=O)N1 c1(C(=O)NC(CN(CC(=O)NCC)CC)C)cc2c(cc1C(=O)NC)NC(=O)C2 C1(C(=O)NCC(C)(C)C(F)(F)F)CCCN1NC(=O)C1(C)CCCC1O C(C(=O)NC1CC(CCNC(C2(CO)COC2)=O)C1)(C(C)C)c1cnc(C)s1 CC1CN2CCN1CC2C(=O)NC1CC(O)C1 C(CNC(C1(C)CC1(F)F)=O)(C(C)(C)C)NC(c1c(CC)csc1)=O c1(C(=O)NC(C)CCCNC(C2(C#N)CCC2)=O)cnn2cccnc12 c1(C(N2CCC(CNc3c(C)nc[nH]3)CC2)=O)cccc2c1CNC2=O C1(CC(=O)N(N(CC(=O)OC)CC)CCCC(C)O)CCCCC12CC2 c1(CCNS(=O)(=O)c2cn[nH]c2)ccc2nonc2c1.c12ccccc1N2 C1(CCNC(c2c(CC)con2)=O)CCN(C(c2cc(OC)ccn2)=O)C(C)C1 C1(C(=O)NC(C)CCN(C)C(c2ncc[nH]c2=O)=O)(CC)CCNC1=O N1(C(C2(C)CC3CCC2C3)=O)CCC2(CCCN(C(=O)CCS(C)(=O)=O)C2)C1 c1(NC(=O)NCC(C)N(CCCCCCCC)C)cc(F)cc2nccnc12 N1(C(COCCC=C)=O)CCC(NC(=O)C(C)(C)CNC(C)=O)C(O)C1 N1(C(C2(CNC(C34CC(F)(C3)C4)=O)CCCO2)=O)CC2OCC(CO)C2C1 c1(NC(=O)NC(C)C(C)n2cccn2)cc(C(N)=O)ccn1 C1(NC(c2c(C)csc2)=O)CCN(C(=O)CCOc2ccc(Cl)c(F)c2)CC1C C(c1ccccc1)=CC(=O)NC1C(CNC(c2csnn2)=O)C1.C1(CO)(N)CC1 CCC(C(=O)NC1(CO)CCCN(c2nccc(-n3nc(C)cc3C)n2)C1)C(C)O N12CC3(C1)CN(C3)C(=O)c1cccc(c1)C2=O.c1(NC(=O)OC)ncccc1F C1(CC)CCCC1C(=O)NCc1occc1C(=O)N(C1CCOC1)C1CC1 c1(C(=O)NCC2CCN(C(CC3(COC)CC3)=O)C2)nn(C)cc1Br N1(C(C(C)=CC2CC2)=O)CCCCC1CC(=O)NCCCCC(C)C Cc1onc(CC(N2CC(NC(=O)CN(C)C(=O)C3CC3)CC(C)C2)=O)c1C#N C(c1ccc(Cl)cc1F)=CC(=O)NCC(C)N(C)C(C1CC(C)CO1)=O C(c1cn[nH]c1)=CC(=O)N(C(C)CNC(C1CCCN1C(=O)OC(C)(C)C)=O)CO CCC(C)CC(C)C(=O)N1CC2(NC(=O)C(=O)NC3CC3)CC1C2 N1(C(CCCCC#N)=O)CCN(C(=O)COC2CCCC2)CC(CO)C1 C1(NC(C(CCC)N(C)C)=O)CCC2CN(C(c3cncnc3C)=O)CC2C1 c1(C(=O)NCC(c2n(C)ncc2)O)ccc(S(=O)(=O)N2CCOCC2)o1 c1(CC)cccc(C(=O)N(CCCN(C(=O)CCN2CCCOCC2)C)C)c1N N1(C(c2c(CC)nns2)=O)CCC(C)C(NC(=O)C(C)Oc2ccc(C)cc2)C1 N(C)(C1c2ccccc2CC1O)C(c1oc2ccc(OC)cc2c1)=O c1(C(N2CC(C)N(C(C3CC(C)N(C)C3)=O)CC2)=O)ccc2nn(C)cc2c1 CC1ON=C(C(=O)N2CC3(CNC(C4CC(N(C)C)C4)=O)CCC2CC3)C1C c1(C(C)NC(C2CCCOC2)C)ccc(-n2cccn2)cc1 C(=O)(C(C(C)(C)C)NC(=O)C1=C(C)CC1)Nc1cc(SC)oc1 N1(c2c(C(=O)OC)ccc(O)n2)CCC2(CCN(C(=O)CC34CCCC3C4)C2)C1 c1(C(N2CC(NC(=O)OCC)C2)=O)cc(C(F)(F)F)ccc1C.C1(=O)C(CN)N1 C#CCC(C(=O)NCCCCCCO)NC(=O)CCC1CCCN1C=O C1(O)(CC(N2C(CNC(c3c(OC)ccs3)=O)CC2)=O)CCCN(C)C1 c1(N2CCCC(CC)(CO)C2)nc(NCC2CCCOC2(F)F)nc2c1CCC2 C1(C)(C(=O)NC(CC)CNC(=O)CC2CCSC2)COCCO1 Cc1[nH]nc2cc(C(=O)NCC(c3ccccc3)CNC(=O)C(C)O)ccc12 C1CC(C(F)(F)F)C1.CC(Cn1ccnc1)C(=O)N(C)C CCCN=C(NCCc1cc(F)ccc1C)N1CCc2c(C(C)C)cccc2C1 Cn1nc([N+](=O)[O-])cc1C(=O)NC(CNC(=O)CCOC1CCCCC1)CO C1(CC(N2CCC(O)(C(=O)O)C2)=O)CCCC(F)(F)C1.C12(CCC1)C(=O)NC2 O=C(N=c1[nH]oc2cccnc12)C1CC2(CC2)CN1Cc1ccc(O)cc1F CCCC(C(=O)NC(CO)C(=O)NC(C)CCC)OC C1(C(N2CCCC(N(C)CC)C2)=O)CC2OCCC2N1 CC(C)C(CNC(c1c[nH]c(=N)o1)=O)C(=O)NC(c1ccccc1)CF C(=O)(C(C)S(C)(=O)=O)N1CC2C(N(C(c3cc(OC)n(C)n3)=O)C)C2C1 C(=O)(C(COC)N(C)C(c1c[nH]c(C)c1)=O)NC1(C(=O)OCC)CCC1 C1(C(=O)NCCCCCC)CC(O)CCN1C(=O)CCC1CC(C)C1 CC(C)CC(C)C(=O)NC1CCCC1CNC(=O)CSc1ccncc1 N1(C(c2cn(C(C)C)nc2)=O)CCC(=CCNC(C2(C)CCC(C)C2)=O)CC1 C(=O)(C1CNC(=O)c2ccccc21)N1CC=CC(NC(COCCCC)=O)C1 Cn1cc(C(=O)NC2COCCN(C(c3n[nH]cc3C3CCC3)=O)C2)n(C)c1=O C1(CC(=O)NC2CC(CNC(=O)CC3OCCO3)C2)CCCSC1 N1(C(c2c(COC)scc2)=O)CCC(CCOC)(NC(c2cc(C)[nH]n2)=O)C1 C1(C)(n2cc(CSCC)nn2)CCCN(C(=O)CNC2CCCC(C)C2)C1 c1(C2(CNC(C=C)(C)CC)CC2)cccc(Cl)c1OC C1(C(=O)NCC(C)NC(=O)CSc2ccccc2)CCC2(CCC2)OC1 C1(C(=O)NC2C3(NC(C=NOC)=O)CCC(C2)C3)CC(F)(F)CCC1(C)C C(=O)(C(CCOCC)NC(=O)CC1CC=CC1)NC(CC#C)(C)C C=CC(CCC)CC(=O)NC1CCCC1NC(=O)CCc1ncc[nH]1 N1(C(CCC#C)=O)CCC2CCN(C(c3nc(-c4cccs4)oc3C)=O)CC2C1 C1(CS(=O)(=O)NC)CCCN(N2CCC(c3ccco3)CC2)C1 CC1(C)CCC=C1C(=O)NCCNC(C1CC2(C1)CC(F)C2)=O N1(C(C2(COC)CC=CC2)=O)CCN(C(=O)CC(C)(C)C2CC2)CC(C)C1 Cn1nnc(CNC(c2cnsn2)=O)c1C(=O)NCCn1cnnc1 C=C1CC(C)(C(=O)NCC=CCC(=O)Nc2cnn(CC)c2)C1 Cn1nnc2cc(C(N3CCC(C)(C)C(NC(=O)CCS(C)(=O)=O)C3)=O)ccc12 c1(NC(N2C(CCC)(COC(C)=O)CCC2)=O)ccc(CC)c(C)c1 C(c1cccc(C#N)c1)=CC(=O)N(CC(C)NC(=O)CC1CCCSC1)C c1(C(N2C(C)(CNC(C3CC=CCO3)=O)CCC2)=O)cc2ccccc2s1 C1(NC(c2cnc(C(C)(C)C)nc2)=O)CC2CC1N(C(c1cocn1)=O)C2 CCCC(C)CC(=O)NC1(CNC(c2cc(C3CCC3)nn2C)=O)CCCC1 C1(NCC(S(=O)(=O)N(C)CC)C)N(C(=O)OC(C)(C)C)CCC1(C)C C1(C(=O)NCC=CC(N2CC(CC)(OC)C2)=O)CN(C)C(=O)N1 C1(NC(c2c(CC)c[nH]c2)=O)CN(C(=O)C(C)(C)c2cnsc2)CC1C c1(C(CNC(C(C=C)C)=O)NC(c2cc(COC)[nH]n2)=O)ccc(C)cc1 N1(C(C(C2CC(NC(CCCC=C)=O)C2)F)=O)CCC(C2CCOC2)C1 N1(C(c2nnn(C)n2)=O)CCN(C(c2cn(C)c(=O)n2C)=O)CC(O)C1 C1(C(N2C(CCNC(C(C)=CC(C)(C)C)=O)CSCC2)=O)CCC(C2CC2)C1 C1(C2C(C(=O)NC(C)Cc3cc(CN)on3)C2)CCCCN1 C1(O)(CNC(COCCN(C)C)=O)CC(NC(c2coc(C(F)F)c2)=O)C1 c1(CNC(C2CC3CCC2C3)C)nc2cc(Br)ccc2o1 CCC(C(=O)NCC(CCOC)NC(=O)C=CC(F)(F)F)n1nccc1C C1(C(C)NC(=O)C(O)CC2CC2)CCN(C(=O)C(c2cccn2C)=O)CC1 N1(C(C2(c3ccc(C)cc3)CC2)=O)C2CCC1CN(C(=O)C1=CCCOCC1)C2 C#CCC(C)(C(=O)N(CCC(=O)NC1CC=CCC1C)OC)OC C1(NC(C(C)=C2CCCC2)=O)CCC2CN(C(=O)C(C)CC3CCC3)CC2C1 CC1C(NC(c2cc(S(N)(=O)=O)co2)=O)CC2CCC1N2C(=O)Cn1ncnn1 N1(CCNC(C(CSC)NC(=O)CC=CC(C)(C)C)=O)CCOCC1C c1(OCCC(N2CC(C(C)NC(C3CC3(C)C(F)F)=O)C2)=O)ccccc1F c1(C(N2CC(F)(CNC(=O)C=CSc3ccccc3)C2)=O)cncc(F)c1Cl c1(C(=O)NC2C(C)CCN(C(CCN(CCC)C)=O)C2)cnc2cccnc2c1 c1(N(C(C2N(CC)CCC2)=O)Cc2ccc(C#N)s2)ccc(Cl)cc1 CCC(CCCC(=O)NCCCSC)NC(C1CCOC1(C)C)=O N1(Cc2c(OC)c(Br)ccc2)CCCC2CN(C3CC3)CCCC12 Cc1ccc(CCC(=O)NC2CC(NC(C3COCCO3)=O)C2)s1 C(=O)(C(O)P(C)(C)=O)N1C(C(CNC(c2nc(C)nn2C)=O)(C)C)CCC1 C=CC(CCC)CC(=O)NCCC(C)(C)CNC(=O)Cc1cc(C(F)(F)F)co1 c1(OCC(=O)NCC(C2COCCO2)C2CCC2)cccc(C2CC2)c1 Cc1nn(C)c(C)c1S(=O)(=O)N1CC2CC1CN2C(=O)CC(C)(C)C C1(NC(C2(CC=C)CCN(C(=O)Cc3ccn(C)c3)C2)=O)CCCCC1CCC C#CC1CCCCN1CCc1ccc(Br)cc1Cl C12(C(=O)NC3CC(NC(CCC(=O)NC4CCCC4)=O)C3)CCCC(C1)OC2 C(=O)(CC1C(=O)Nc2ccc(F)cc21)NCC=CCNC(C(C(C)C)(C)C)=O CCCC(C)C(C(=O)NCCn1cc(-c2ccnc(F)c2)nn1)N1CC(CC)C1 C1(NC(COCc2onc(C)n2)=O)CCN(C(c2coc(C(F)F)c2)=O)C12CC2 C(N=c1[nH]c(N2CC=C(C)C2)nc2cc[nH]c12)c1cccc(OC)c1 c1(OCC)ncc(NC(=O)C(c2cncn2C)O)cn1 N1(C(c2ccc(C)o2)=O)CCC(C)(C)C(CNC(c2ccccc2)=O)C1 CCCC(C)(C)CC(=O)N1CCN(C(c2ncoc2Br)=O)C2CC12 c1(C(N2C(COC)CN(C(=O)CCC3CC3)CC2)=O)onc2cc(C)ccc12 N1(C(=O)CCn2cc(C3(O)CCCC3)nn2)CC=CCC1CO N1(C(c2c(C)cnn2C)C(=O)NCc2ccc(F)cc2)CCN2C(=O)NC(=O)C2C1 CC1(C)CC(NC(C2(C)CCN(C(=O)CC3CCCC3O)C2)=O)CC(O)C1 c1(OC)cc(O)ncc1C(N1CCC(CC(C)NC(c2cc(O)cs2)=O)CC1)=O C(=O)(C(C)(C)CC1CCCO1)NCC1(NC(CC(=O)NCC)=O)CCCC1 c1(C(=O)NCC2CC(NC(C3CN(C)C(=O)N3)=O)C2)ccc2c(c1)COCO2 c1(C(N2CC(NC(c3cc(C)no3)=O)(CO)C2)=O)cc(N2CCCC2)nc(Cl)c1 c1(C(=O)NCC(=O)N(C)Cc2cn(CC)nc2)ccc(O)nc1C C1(CCNC(N(C(C)C)Cc2coc(CO)c2)=O)CCOC(C)C1 c1(COC(CCc2snc(CC)n2)=O)cccc(C(F)(F)F)c1 c1(C(=O)NC2C(C(N(CCCCCC=C)C)=O)CCC2)c(F)cc(Br)cc1Cl c1(CC)cc(CC(=O)NC(C2(O)CN(C(=O)C(c3cnn(CC)c3)=O)C2)C)on1 N1(C(C=CC)=O)CCCC(CN(C)C(c2ccsc2OC)=O)C1 CC1=C(C(=O)NC2CCC(N(C(=O)CNc3cccnc3)C)C2)COCC1 N1(CC(=O)NC2CCCC2)CC2CCC1C1CN(C(=O)Nc3ccnc(F)c3)CC21 n1(-c2cccc(C)c2)cc(S(=O)(=O)NC2(C(=O)O)CC2)cn1 O(N(CC)C(=O)C1(c2nnnn2CCNc2cc(Cl)cn2C)CC12CCC2)CC C1(NC(CC2CCN(C)CC2)=O)COC2(C1)CN(C(=O)CCC1CC(F)(F)C1)C2 c1(C(=O)OC)cc(C#N)cnc1N(CCCNC(c1nc(C)ncc1Cl)=O)C Cc1cc(=NC(=O)C(=O)N2CCN(C(=O)CC)CCC2C)[nH]o1.N1CCCCCC1 C(C(C(=O)NCc1cnn(C(C)C)c1)C(C)C)NC(CC(C)OC)=O C1(CN(C)C(C2CCC=CO2)=O)CCCCN1c1nnc(C(C)(C)C)o1 C(C(O)CC(=O)NC(c1ccco1)CO)NC(CCCSC(C)(C)C)=O CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(c3cc(Br)no3)=O)C2)C1=O C(=O)(C(CC(=O)OC)OC)NCC1C(NC(COCCOCC=C)=O)CCC1 c1(OCC#C)ncccc1C(=O)NCC1(CCNC(=O)Cc2ccccc2)CC1 C#CC1CCN(C(C2OCCC2NC(C2CCC3(CC3)C2)=O)=O)CC1 N1(C(C2CC23CCN(C(=O)C(F)C(F)(F)F)C3)=O)CCC2(CCCO2)C1 C1(NC(c2cc(CSCC)on2)=O)CCCC12CN(C(=O)CC1(CO)CC1)C2 N1(C(c2c(Cl)cn(CC)n2)=O)CCCN(C(c2ccsc2)=O)C(CO)C1 c1(C(=O)NC(CNC(c2cn(C)nn2)=O)C2CC2)cnc(Cl)cc1Cl C1(C(N(C(C)CNC(=O)CC(c2cccs2)C2CC2)C)=O)CCCCC1(C)C c1(OC)cc(-c2ccc(NCc3cccc(Br)c3I)nc2)ccc1C n1(CC(=O)NCC(C)NC(C2CC3CCC2O3)=O)cnc2ccc(F)cc2c1=O C1(C(N(C2(C#C)CC2)CC)=O)CCN(C(=O)CC2CCCC2)C1(C)C Cc1cc(C(=O)NC2(C(N3CC(O)C(O)C3)=O)CC2C)nc(C)c1 N1(C(C2(CCOC)CCC2)=O)CCC(C)(CNC(C2CCCCC2O)=O)C1 C(=O)(C1CCCn2nccc21)NC(C)C(CO)NC(c1ccc(Cl)cn1)=O Cc1cc(NC(=O)C(O)C2CN(C(C3C4CN(C)CC34)=O)C2)c(O)c(C)c1 C(=O)(C1=NN(CC(C)C)C(=O)CC1)NCC(C)N(C(=O)COC)CC CC(O)(CC(=O)N1CCC2C(CCN2C(c2ccnnc2)=O)C1)C(F)(F)F C#CCCCCCC(=O)NC1CCCC1NC(c1cc(Cl)c[nH]1)=O N1(C(CC=CCC)=O)CCCC1C(C)NC(C1(C(F)F)CCCO1)=O N1(C(C(COC)OC)=O)CCCCC1CNC(C1(CSC)CC1)=O c1(C(=O)NCCNC(c2nn(C)c(C3CC3)c2)=O)cc2c(F)c(F)ccc2[nH]1 C1(NC(COC)=O)CCCOC12CCN(C(=O)C(C(C)C)n1cnnn1)CC2 c1(C(=O)NC2CC(NC(C3CC4C=CC3O4)=O)C(O)C2)cnc2c(c1)CCOC2 c1(C(N2CC(C(C)C)N(C(c3cccnn3)=O)CC2)=O)ccc2c(n1)NCC2 C1(CC)CN(C(=O)C(=O)NCCF)CCN1C(=O)Cc1cc(C)n(C)n1 c1(C(=O)NCC2CN(C(c3ncn(-c4ccccc4)n3)=O)C2)cc2sccc2[nH]1 Cc1cccc(C2C(C(C)Nc3cccc(OCc4nn[nH]n4)c3)C2(C)C)c1 C(C(F)(C(=O)NCC12CCCCC1C2)C(C)C)NC(C(C)=CC=C)=O CC1(C)CCCC1C(=O)NC(C1CCCC1)CNC(c1ccc(Cl)s1)=O CC1CC2CCN1c1nnc(Cc3cncc(F)c3)n1C2.C(C)(C)(C)SC C(=O)(CC1CCc2ccc(O)cc21)N1C(CCNC(=O)CCCF)CCC1 C(=O)(C#CC1CCC1)NCC1CN(C(c2cnn(CC)c2C)=O)CC1C(F)(F)F C(C(=O)N(C)CC1(C#N)CCC1)(C(C)O)NC(CCC=C(C)C)=O N12CCC3CCC(CC13)C2=O.c1(C(=O)OC)ccc(C2CNCCO2)cc1 N1(C(C(F)=CC)=O)CC(O)(C2CCN(C(=O)Cn3cnc(C(F)(F)F)c3)CC2)C1 N1(C(=O)C(c2ccc(F)cc2)=O)CCCC2C1CCCN2.C1(N)CCOCC1 c1(NC)cccc(C(N2CC(C)(C)C2C2CCN(C(=O)C=CCOC)CC2)=O)n1 N1(C(c2cnc(COC)s2)=O)CCN(C(=O)C(C)(C)N2CCCCC2)CC12CC2 c1(N2CCN(CC#CC)CC2)nc2c(c(=NCCc3nccc(C)n3)[nH]1)CSC2 O=S(=O)(c1ccc(NC2CCC3CCC23)cc1Cl)NCCSCCO N1(CC)CCC(NC(=O)C(C)(CSC)NC(c2cc(O)nn2C)=O)C1=O CC1CN(C(=O)CC2CC=CCC2)CC1NC(=O)COc1cccnc1 C1(CCCNC(C=CC(C)C)=O)CCN(C(C2C=CCS2)=O)CC1 C(c1nc2ccccc2o1)=CC(N1CC(NC(C2CCC(CCC)CC2)=O)C1)=O C1(NC(C2N(C(N)=O)CCCC2)=O)CN(c2ncc(Cl)cn2)C2(CCOCC2)C1 C1(C(=O)NC2CN(C(C)C)CC2C)CCC2CCC1N2C(c1cn(C(C)C)nn1)=O N1(c2cc(C(=O)OC)ncn2)CC2CCCC(CNC(=O)CC(F)(F)F)C2C1 N12CCC(C)(CC1)C2=O.C1(C(=O)OCC)CCCN(C(=O)NC)C1 C1(CNC(C2CC(CC)C2)=O)CCC2(CO1)CC(NC(=O)C(O)C1CC1)C2 c1(NC(CNC(C2(COC)CC2)=O)=O)ncc2ccccc2n1 c1(OC)ccc([N+](=O)[O-])cc1C(N1CC(C(C)NC(C2CC(N(C)C)C2)=O)C1)=O c1(C(C(=O)NC(c2cccc(C(F)(F)F)c2)C)(C)N)ccc(F)c(Cl)c1 c1(C(N2C(C=C)COCC2)C(=O)NCC2CCCO2)cc2ccccc2o1 c1(C(=O)NCC2C(C)C2(F)F)ncc(N)cc1Cl O=C(CCCNCc1ccc(Cl)nc1)N=c1cc[nH]cc1 N1(C(c2cccc(C)c2)C(=O)NCC2CCOCC2)CCCC2OCCC2C1 N1(CC(N2CC(CC)(NC(=O)CCCC(C)C)C2)=O)CCn2ccnc2C1 C1(NC(c2ncc(C)cn2)=O)CS(=O)(=O)CC1NC(c1ccc(F)cc1C)=O c1(CC(=O)NCC2CC(NC(C=C3CCC(C)C3)=O)C2)cc(Cl)sc1Cl N1(C(Cn2ncc(C)c2)=O)CCCC2C1CCN2C(=O)C(=O)N(C)C CC(C)CC(O)CN=c1ccc(Br)c(S(=O)(=O)NCCC(C)N2CCCC2)[nH]1 c1(CC(N2CC(NC(c3ccc(COC)cc3)=O)C2)=O)cc(F)cc(F)c1F C(=O)(C(C)CC(F)(F)F)NCC1C(NC(CCC(=O)N(CCC)C)=O)CCC1 c1(C(=O)NCCC(C)(C)NC(c2c(CC)n(C)cc2)=O)cc2c(s1)CCC(C)C2 c1(CC(=O)NCCC2(OC)CN(C(c3cc(F)c[nH]3)=O)C2)nc(F)c(F)cc1F C(=O)(C#CCNC(=O)C=C1CCCCC1)NC(C)Cc1cn(C)cn1 c1(NCC2CN(C)C2)ccc(S(=O)(=O)NC2CCC(n3ccnn3)CC2)c(Cl)c1 Cc1ccc(C(=O)NC2COCC2NC(C2(C(F)(F)F)CC(F)(F)C2)=O)cc1Cl C(=O)(CCC(=O)N1CCOCC1)NCC(CN(C(C1N(CC)CC1)=O)C)C c1(C(=O)NCC2(OC)CN(C(=O)C=CC(N)=O)C2)cnn(-c2ccccc2)c1N N1(C(c2ccc(OC)cn2)=O)CCN(C(c2ccnc(CO)c2)=O)C2CCCC12 N1(C(C=CCNC(CCc2n(C)cnn2)=O)=O)CCOC2C(O)CC12 N1(C(C(C)(C)SC)=O)CCC2(CO)CN(C(=O)Cn3nc(O)ccc3=O)CC2C1 N1(C(CCSC)=O)CCN(C2CCCN(C(C3(C)CCCS3)=O)C2)CC1 C(=O)(C(CNC(c1ccnn1CCF)=O)C(C)C)NCCC(C)OC CC(C)C(C(=O)N1CC(=C(F)CNC(C23CCC(CO2)C3)=O)C1)N(C)C C1(NC(c2cc(OC)cc(Cl)c2)=O)CC2CC1CN(C(=O)C1=C(C)OCCS1)C2 N1(CC)CCC(Nc2ccc(C(=O)NCC=CC(OC)OC)cn2)C(C)C1 c1(C(N2CC(CC(=O)NCc3c(Cl)ccc(O)c3Cl)C2)=O)cc(Cl)c(Cl)nc1Cl CC1CCC(CNC(=O)CCc2nc[nH]n2)N(C(c2ccnc(O)c2)=O)C1 c1(CCC(=O)NCC2C3CN(C(CC4ON=C(C)C4)=O)CC32)c(F)cccc1F N1(C(CC(CCC)(C)O)=O)CCCC(C2CN(C(=O)C(C)CN(C)C)C2)C1 N1(C(CC(C)F)=O)CC(CNC(c2cnn(CCO)c2)=O)OC2COCC12 N1(C(C(CC)(CC)CC)=O)CC2CC(C1)CN(C(c1ccnc(N(C)C)c1)=O)C2 c1(C(=O)NCC2C(C)CN(C(c3ccoc3Cl)=O)CC2)cnn2c(N)ccnc12 N1(C(CC(C)SC)=O)CCC(=CCNC(=O)CCCN2CCCCC2)CC1 C(CC(=O)NCCNC(=O)C(C)(C)C1CCCCO1)(C1CCCC1)NC(C)=O C1(NC(c2cccc(CC)n2)=O)CN(C(=O)C(c2cccc(C)c2)F)C(C)(C)C1 c1(C(N2CCC(C(C)NC(=O)Cc3ccc(Cl)cn3)C2)=O)cn(C)c(=O)n1C c1(C(N2CC(NC(C(c3ccccc3)C)=O)C2)=O)cccc2c1NC(=O)CC2 N1(C(COCC#C)=O)CC(F)(F)CC1CNC(=O)C(C)n1ccnn1 c1(C(=O)NC(CCCNC(c2cccc(OCC)c2)=O)C)ccc2ccnn2c1 c1(C(N2C3CN(C(C4CC4c4ccc(O)c(O)c4)=O)CC32)=O)ccc(O)c(I)c1 C(=O)(CCC(F)F)N1CC(CNC(C(C)C2CCCC2)=O)C1 C1(CC(=O)NCC(N(C)C(c2cnc3n2CCS3)=O)C2CC2)CCC(C)(C)CC1 c1(CC(=O)NC(C(CO)NC(Cc2c(C)nc[nH]2)=O)C)ccnc(Cl)c1F c1(OCC(N2CC(c3cn(CC(F)(F)F)nn3)C(O)C2)=O)ccc(F)cn1 C1(C(N(C)CCc2ccc(F)cc2)=O)CC2CCN(c3ncccc3CO)CC12 c1(CC)ccc(NC(=O)C(CN(C)C)NC(=O)C(c2cncnc2)C)c(C)n1 c1(NC(=O)Nc2c(C)nc(CCC)s2)c(C)cccc1Cl C(C(=O)NOCC1CCCO1)(C1CCOC1)NC(c1c(CC)nn[nH]1)=O Cc1nc2cc(C(N3CCC3CNC(C3CCCC(C)(C)C3)=O)=O)ccc2o1 O=C(C1COc2ccccc21)N1CC2CC(C1)C2NC(C1(Br)CC1(F)F)=O N1(CCCC)C(CNC(C(C)NC(=O)OC)=O)=CC=C(F)C=CC(S)CN(C)C1=O C1(CCCN(C(C2(CCl)CCOC2)=O)CCO)CCCN1c1ccccc1 C1(NC(C(CC)=CC)=O)CC2CC1CN(C(=O)CCCn1nc(C)nc1C)C2 N1(C(CC(=O)OCC)=O)CCCC(F)(C(=O)NC2(C)CCOCC2)C1 C(CCCCCCCN(C)C)NC(CCC)CCCO.C1C(=O)N1 CC(C)C(C)(CNC(C1CC=CCC1)=O)NC(=O)CCc1cncnc1 n1(C(C)C(N2CCN(C(=O)CCc3ccon3)CC2)=O)cnc2ccccc12 C1(NC2C(C)CN(C(=O)OC(C)(C)C)CC2)(CO)CCC2(CCOCC2)C1 CN1CCC(CC(=O)NCC2CCCCN2C(c2cc(Cl)c[nH]2)=O)C1=O c1(OCCOC)cccc(NC(C2CC(C(=O)O)C2)=O)c1 N#Cc1cnccc1CNC1CCN(C(=O)COc2cccnc2)CC1O C1(CNC(COCC(C)C)=O)CN(C(c2csc3nccn23)=O)CCCO1 C1(C(F)(F)F)(C(=O)NCC(CN(C(COC)=O)C)O)CC2C=CC1CC2 C1(C(N2CC(O)(CCNC(=O)C(=Cc3c[nH]cn3)F)C2)=O)CC2CCC1CC2 Cn1cc(C#CCNC(c2ccc(CNC(c3ccc(F)cc3F)=O)nc2)=O)cn1 CCC(CC(=O)NCC1(O)CN(C(C2CC(F)(F)CCC2(C)C)=O)C1)C(C)(C)C N1(C(c2cc(C)c(C)nn2)=O)CCC2(CC1)CC(NC(C1C3CCCC13)=O)C2 c1(C(N2C3CN(Cc4c(C)cc(Br)cc4C)C(C3)C2)=O)c(Cl)ccc2c1OCO2 C12(C(N3CCC(C(C)NC(=O)CC4CC5CC5C4)C3)=O)CC3CC1C2C3 C=CCC(C)C(=O)NCCC1(CNC(=O)CCSCc2csc(C)n2)CC1 c1(C(=O)NCC(CC=C)NC(C2(C)CC=CCC2)=O)cnc(O)c(Cl)c1 C(C1=NOC2CN(C(=O)CCNC(N)=O)CC12)NC(c1c(CC)onc1C)=O c1(C(=O)NC(C2CCCC2)CNC(=O)Cc2ccco2)scnc1C(F)(F)F C1(NC(c2cnc(SC)s2)=O)CC(O)CN(C(=O)CCCSC2(SC)CCC2)C1 C=CC(C)(O)CC(=O)N1CCC1Cn1cc(CCCN2CCCC2CO)nn1 CC1CCCC(O)(C(N2CC(CCNC(C3(F)C(C)(C)C3(C)C)=O)C2)=O)CC1 C(=O)(C(F)(F)CO)N1C(C2(N(c3nc[nH]n3)C(=O)CN3CCCC3=O)CC2)CCC1 c12cncc(c1)NC2.C1(C(N(C(C(C)OCC)=O)C(C)C)=O)CCC(N(C)C)C1 n1(CC)cc(NC(=O)C=CC2CCCN2C(=O)CCCC2CCCO2)c(C#N)n1 Cc1ncc(C(=O)NCC2(NC(=O)C(C)NC(=O)CNC(N)=O)CCCC2)o1 C1(NC(=O)CN2CCCS2(=O)=O)CCCCCN(C(C23COCC2C3)=O)C1 C1(C(C)NC(c2c[nH]c(Br)c2)=O)CCCN(C=O)C1.c1cscn1 c1(C(=O)NCC2(C)CCN(C(=O)CO)C2)ccc(Br)c2cn[nH]c12 N1(C(c2nc(C)[nH]n2)=O)CC2CC1CN(C(=O)CC1OCCC1(C)C)C2 c1(C(N2CC(NC(C=COCC)=O)C3C2C3)=O)ccc(N2CCC(C)=N2)cc1 N1(C(CCOCCOCC)=O)CCN(C(=O)Cc2ccc(Cl)c(F)c2)C(C)C1C c1(-c2cccc(NC(=O)CC3CCCCO3)n2)cccc2ccoc12 N1(C(CCC#C)=O)CCCC(NC(=O)Cc2c(C)nn(C)c2Cl)C(F)C1 C1(NC(CCc2scc(C)n2)=O)C2CC1N(C(c1ncoc1C1CC1)=O)C2 c1(C(=O)NC(C2(O)CCN(C(CCC(C)C)=O)C2)C)ccc(F)c(Br)c1 C1(NC(CCOCCCNC(C(C)C)=O)=O)CN(C)NC1=O C1(C2=CCCCCC2)(C(N2CC(C3N(C(CSCCC)=O)CCC3)(O)C2)=O)CC1 c1(C(=O)NC(CCOC)CNC(=O)C(C)n2cccn2)cc(N)ccn1 c1(CC(N2CCOCC(CNC(C(C)=C(C)C)=O)C2)=O)cccc2sccc12 c1(OC)ccc(C(C)C(=O)NCC2(CO)CCCO2)c(C)c1 C1(CN(C(C(CC)OC)=O)C)C2CN(C(=O)C=CC=C(Cl)Cl)CC12 c1(C(=O)NCC(C)N(C)C(c2cc[nH]c2C2CC2)=O)cc2c(F)ccc(F)c2[nH]1 c1(C(=O)NC2(C)CN(C(c3ncn4c3CCC4)=O)C2)nccn2cnnc12 N1(C(c2cc(SC)oc2)=O)CCC(CNC(=O)C2=CCSC2)C1(C)C c1(C(=O)NC2CCC(N(C)C(c3cc(CF)on3)=O)C2)n[nH]c2c1CCOC2 C1(CNC(c2nc(C)oc2)=O)CN(C(=O)C2=CSCS2)CC1C(F)(F)F C(=O)(C1=C(CCl)N(c2ccc(Cl)cc2)C(=S)NC1c1ccc(C)cc1)OC Cc1sc(S(N)(=O)=O)cc1C(=O)NC1CCC1CNC(=O)CCOC(C)C N1(C(C(C)=O)=O)CCCN(C(=O)C(C)NC(c2cccc(C)c2)=O)CCC1 C1(NC(COC)=O)CCC2CCN(C(C3(C)CCCC3)=O)C12 c1(C(N2C(C(C)(C)NC(C3CC(N=[N+]=[N-])C3)=O)CCC2)=O)ccc(S(C)(=O)=O)o1 c1(C(N2CC=CC(NC(C3C(C=C)CC3)=O)C2)=O)ccc(C)c(CC)c1 c1(CC(N2C(CNC(CCSCCCC)=O)C(CC)CC2)=O)c(O)cccc1F c1(NC(N(CC(=O)OC(C)(C)C)C)=O)ccc2c(c1)CCC1(CCC1)O2 N1(C(C(C(C)C)NC(C)=O)=O)Cc2[nH]nc(C(=O)NCC3(S(C)=O)CC3)c2C1 c1(C(=O)NCC(C)(C)NC(c2cc(F)c[nH]2)=O)cc2occ(Br)c2[nH]1 c1(C(N(CC(C)NC(=O)Cc2ncc(C(F)(F)F)[nH]2)CC)=O)cn2ccnc2s1 N#Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CCC2NC(=O)Cc2ccoc2)c1 C1(C(=O)NC2(C#N)CCN(Cc3c(OC)cccc3Br)C2)Cc2ccccc2O1 C1(NC(=O)Cc2cc[nH]c2)CCCC(CO)C1.C12C=CCCC1C(=O)N2 C=CC1(C(=O)NCCN2CCOCC2C)CCN(C(=O)CCC(C)(C)OC)C1 C(=O)(C(C)CCC(C)(C)C)NC(CCOCC)C(=O)NC(CC)C1CCC1 c1(OC(C(=O)NCCC(=O)N(CCOC)C)C)cc(F)cc(F)c1 Cc1cc(Br)c(F)cc1C(N1CCC(O)(C(=O)Nc2cnccc2Cl)C1)=O c1(C(=O)NCCC2CCCN(C(c3cc[nH]n3)=O)C2)cc2c(F)cc(F)cc2[nH]1 C1(NC(c2cn(CCOC)nc2)=O)CN(C(C2CC2(F)F)=O)C2(CCOCC2)C1 C12(C(N(C)CC3C4CN(C(c5sccc5Cl)=O)CC34)=O)CCCC(=O)N1CCC2 C1(CC)C(NC(=O)C(O)P(C)(C)=O)CCCN1C(=O)COCC1CCOC1 N1(C(C2CC(SC)C2)=O)CCN(C(c2cnn(C)c2)=O)C2CS(=O)(=O)CC12 N1(C(CCCOCC)=O)CC2CCC1C1CN(C(=O)C(C(C)C)OCC)CC21 N1(C(c2ccc(OCCF)cn2)=O)C2CCC1CC(NC(C13CC(O)C1C3)=O)C2 C=CCN=c1nc(N2CCN(C)CC2)c2ccccc2[nH]1 N1(C(C2(C)COC2)=O)Cc2ccccc2C1C(=O)Nc1cccc(Cl)c1CO N1(C(c2n(CC)ccn2)=O)CC(NC(=O)CC2CC(F)C2)C2CCCCC12 CCCN(Cc1ccc(C#N)cc1)N1CCN(Cc2cccc(C)c2O)CC1 c1(C(=O)NCC(CC)NC(c2cc(Br)cnc2O)=O)ccccc1S(C)=O c1(C(N2CC3C(NC(C=C(C)C)=O)(CC3)C2)=O)ccc(C)c2ccccc12 C1(CCCCNC(c2cccs2)=O)CCCN(CCN(C(=O)C(O)C(F)F)CO)C1 C1(CC(C)(C)C)CN(C(=O)COCC2CCC2)CCN1C(=O)CNC=O c1(CN(CCNC(c2nccnc2-n2ccnc2)=O)CC)cnn2c1CCCC2 N1(C(C2N(C(c3cc(C)c(N)cn3)=O)CCC(F)C2)=O)CC2(CC(CO)CO2)C1 C12(NC(CCNC(COC)=O)=O)CCCC1N(C(C1C(C)(C)C1(F)F)=O)CC2 c1(C(N(C=O)Cc2c(Cl)ccnc2Cl)C)ccc(F)c(Br)c1 C1(NC(Cc2c(C)cco2)=O)CCN(C(c2coc(C3CC3)n2)=O)CC1O O(NC(=O)C1=CCN(C(c2cnc(N)cn2)=O)CC1)CCCOC c1(C(=O)NC2(CNC(C3(O)CCCC3)=O)CCCCC2)cc2c([nH]1)CCCC2=O c1(SC)ccc(C(=O)NC(C)CNC(c2ccc(=N)[nH]c2)=O)cc1Br C1(C(=O)NC2CC=CC2)CCN(C(=O)C2=C(Cl)CCOC2)C12CCC2 c1(C(=O)NC(CCOC)CNC(C2CCCN2C(C)C)=O)cccc(N)c1F C1(N=[N+]=[N-])(C(=O)NC23C(C)OC(CC2)C3)CCN(C(C2CC(=O)CC(=O)N2)=O)C1 N1(C(C2CCN(C)C2)=O)CCC(c2nnc(NC(c3nc(=O)n(C)[nH]3)=O)s2)CC1 C1(NC(COCc2c(C)cccc2)=O)CN(C(c2ccnnc2C)=O)CCC1C C1(C(=O)NCC(C)(C2CC2)NC(=O)CC2(N3CCCC3)CC2)CC(=O)C12CCCC2 O=C(CCC(CF)CF)NC1CCC1CNC(C12CSCC1C2)=O C(=O)(C(C)C(C)(C)C)NCC(CNC(C1(CC)CCOCC1)=O)(C)O C(c1ccc(C(N)=O)o1)=CC(=O)NC1(CNC(C(C)O)=O)CCC1 O(N1C(=O)c2ccccc2C1=O)CC(=O)NC1COCCN(C(=O)CC(F)F)C1 N1(C(c2cnc(CCC)s2)=O)CCC(C)C(CNC(c2nn(C)cc2Cl)=O)C1 C1(C2CCC2)(C(N2CCC(F)(CNC(CCCCOC)=O)CC2)=O)CC1(F)F C=C1COc2c(C(=O)NCCCOCCNC(C3CCC4CC34)=O)cnn2C1 C=CC(C)CC(=O)NCCN(C(=O)C(C(C)C)Nc1ccccc1)C1CC1 c1(NC(C2C(NCc3c(Cl)ncc(OC)c3)CCC2)=O)ccc(C#N)cc1Cl Cc1cnc2n1CCC(C(=O)N(C)CCNC(=O)CN(c1ccccc1)C)C2 N1(C(C=CC(=O)N(C)C)=O)CC2CCC2(CC(=O)N(C2CCCCC2)CC2CC2)C1 CC(C)(CC1CC1)C(=O)N1CCC(CCNC(C2CC3CCC2C3)=O)C1 CC1CC(N(C(=O)CC=Cc2ccccc2)C)CN1C1CC1.C1(=O)CCCN1 C(C(C)(C)C)N(C(=O)CC1CC(CN)C1)CC.c1(C(=O)CC)nc[nH]n1 C(=O)(C(C)C(C)O)N1CC(NC(C(C)C2CCCC2)=O)(CO)C1 C1(NC(C(=O)NCCOCCCC)=O)CCN(C(c2ccon2)=O)CC1 c1(C(=O)NCCNC(C2CN(C(C(c3ccnn3C)C)=O)C2)=O)ncc(F)cc1N C1(C(=O)NCC2N(C(C3CC(OC)C3)=O)C3C(C2)C3)Cc2ccc(F)cc2C1 Cc1cc(C(=O)N(CCCCN(C(=O)C(C)C2CCC2)C)C)n(C(F)F)n1 Cc1nccn1C(C)C(=O)NC1CC(CCNC(C2CC(O)C2)=O)C1 c1(C(=O)NCC2(NC(=O)CCCCN3CCCCC3)CC2)ccc([N+](=O)[O-])cn1 c1(NC(C2CN(C(C(C)n3cccn3)=O)CC2F)=O)nccc2[nH]ccc12 N1(C(C)=O)CCOC(C(N2CCCC(N(C)C(C3(C#N)CCCC3)=O)C2)=O)C1 c1(CCNC(=O)NC(C(F)(F)F)C2CCOC2)cncc2ccccc12 C1(C(=O)NCCC(C=C)C)CC(C)CCN1C(=O)C(COC)N=[N+]=[N-] C(=O)(CCCC(CCC)CCC)N1CC(NC(C(C)OCCCC)=O)C(C)C1 C(CCCCCCO)NC(C1C(CC)CCCC1)=O.N12CC(C)(C1)OCC2=O N1(C(C)=O)CCC(c2ccc(OC)cc2)C(NC(=O)Cc2ccc(O)c(C)c2)C1 C(=O)(CC(C)C(F)(F)C(F)(F)F)NCCN(c1cc(SC)ncn1)CC C1(C(=O)NCCN(CC=C)CC)C=CCOC1 C(=O)(C(F)C(C)(F)F)NCc1cn(C2CN(C(COC(CC)C)=O)C2)nn1 C(=O)(C1CCOc2ccc(Br)cc21)N1C(CCC)CN(C(=O)CC)CC1.OCC O=S(=O)(C1CC12CCC2)NCc1nc(COc2ccccc2)cs1 C12(CNC(C3N(C)C(=O)CCC3)=O)CCCC1CN(C(C1CCCC13CC3)=O)C2 c1(C(=O)NC(C(CC)C)C(=O)NCCc2nncn2C)ccn2ccccc12 c1(C(=O)NCC(CNC(c2cc(C)nc(C)c2)=O)(C)O)ccc2cc(C)cn2c1 c1(NC(=O)NCCN2CCN(CC3CC(=O)N3)CC2)ccnc(F)c1Cl C=CCC(C(=O)NC1CCC(C)N(C(c2ncccc2F)=O)C1)C(C)C N1(C(c2c(CC)cccn2)=O)C(CNC(=O)Nc2cccs2)CC2COCC12 c1(C(N2CCCC(C)(NC(C(C)=CC)=O)C2)=O)ncc([N+](=O)[O-])n1C N1(C(C2C3C4CC5C2C3C45C(=O)N)=O)CC2CCCC(C2)C1.C1(NC)CCCCC1 CC(C)CC(C)CC(C)C(=O)N(CCCNC(=O)Cc1nc([N+](=O)[O-])n[nH]1)C c1(C(N(C2CCCN(C(C=C(CCC)CCC)=O)C2)C)=O)cc(O)nc(C)n1 C(=O)(C(CO)C(F)(F)F)N1CC(CNC(c2c(C)n(C(C)C)cc2)=O)C1 C1(NC(C(Cc2ccco2)NC(c2cc(C)[nH]n2)=O)=O)CN(C)CC12CC2 N1(C(c2ncc(Cl)nc2N2CCCC2)=O)CCC(S(=O)(=O)c2ccccc2)C1 c1(CC)cc(C(=O)NC2(CNC(=O)C(C3CCOCC3)C)CC2)oc1CC C1(C)(C(=O)NC(CN(CC)CC)C)CCCN(C(C2(CF)CC(=O)C2)=O)C1 C1(C(N(C(C)CCNC(=O)C(F)=CC2CC2)C)=O)CC12CCCCCC2 N1(c2nnc(C(CC)(C)C)o2)CC2(CCCC2NC(c2cc(O)nn2C)=O)C1 N1(C(c2c(CC)n[nH]c2)=O)CCC(O)CC1C(=O)NCC(O)C(N)=O CCCC(C)C(=O)NCCOC1CCN(C(c2cnc(C(C)(F)F)s2)=O)C1 c1(CC)cccc(-c2cncc(C(=O)Nc3ncccc3C(C)C)n2)c1F C1(CCC)CN(C(=O)CSc2nncn2C)CCN1C(=O)CP(C)(C)=O N12CCN(CC1)CC2.c1(COC(N2CC(C(=O)OC)C2)=O)ccccc1F C1(CN(C)C(c2ccnc(CO)c2)=O)CCN(C(C2(C3CCCO3)CC2)=O)CC1 CCC(CC)C(C(=O)NC(c1nocc1C(=O)Nn1cccn1)C)OC c1(C(=O)NCc2c(CC)con2)cc(CNC(C2CCCS2)=O)ccn1 C1(NC(CCOCCN(C)C)=O)CC(F)CN(C(=O)CCCc2cnn[nH]2)C1 c1(NC(C2C3(CC3)C23CC3)=O)nc2ccc(Br)cc2s1 CC(C)(N)CC(C1CC1)NCCC1CCCOCC1 N1(C(C(C)O)=O)CCC(NC(=O)C=Cc2cncn2C)CC1C Fc1ccc2c(c1F)C(N)CCS2.N1(c2ccccc2)CCC(c2cn[nH]c2)CC1 c1(OC)ccc(C(N2CCN(C(C3CC=CC3)=O)C(CCO)C2)=O)c(O)c1 c1(C(=O)NC(c2cn(CC3CCC3)nn2)C)ccc2c(=N)[nH]oc2c1 C1(O)(C(=O)NCCC(N2C(C(=O)NC)CC2)=O)CCOC1 N1(C(c2cnc(C)[nH]2)=O)CCN(C(=O)CN2CCN(C3CC3)C2=O)CC(O)C1 N1(C(C(C)O)=O)CCC2(CCCN(C(=O)C=Cc3cccnc3)C2)C1 c1(C(N(C)CC2OCCN(C(C(C)C)=O)C2)=O)nc2n(c1Cl)CCCC2 Cc1c(C(=O)N(CCCN(C)C(C2CC(N(C)C)C2)=O)C)cncc1Br CC1(C(=O)NC(C2CCCC2)CNC(C2CC2C(F)(F)F)=O)CCC1 N(C1CCS(=O)(=O)c2ccccc21)C(c1ccc(F)cc1)CC(C)(C)OC n1(CCCC)nnnc1C(c1csc(C2CC2)n1)NCc1noc(C(F)F)n1 C1(C(N2CCC(F)CC2)=O)CCC(C2CC2)N1C(c1ccccc1CO)=O c1(C(N2C(C(=O)NC3(CC)COC3)CC3CC32)=O)cc(Br)c(C)cn1 Cc1ccc2[nH]c(=NCC(C3CCC3)NC(=O)OC(C)(C)C)sc2n1 N1(C(C2C(CCC)CCC2)=O)CCCC(C)(CNC(c2occc2Br)=O)C1 C(=O)(C1=CC(C)(C)C1)NC(CC#C)C(=O)N(C)Cc1ccnn1C O=S(CCNC1CCOCC1F)c1cc(Br)ccc1F Cc1cc(C(=O)NC(CCF)C(=O)NCC2CN3CCC2C3)oc1C c1(CN2C(c3ccc(C#C)cc3)CCCC2)c[nH]c(=NC2CCCN(C)CC2)cn1 C1(CNC(CC(C)C)=O)CC2(CCN(C(c3ccc(C)c(C)c3Cl)=O)CC2)C1 N1(CCNC(c2cc(OC)ns2)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)CC1 N(C1CCCSc2ccc(Br)cc21)S(C1CC(COC)C1)(=O)=O N1(C(c2cc(C(CC)C)no2)=O)CCC2CN(C(=O)CCC3CCOC3)C2C1 c1(C(=O)NCC(CNC(C=CCC)=O)C)ccc(-n2cncn2)cc1 C(CC(C)C)(C(C(=O)NCc1ccccc1)N1Cc2ccc(CO)cc2C1)OC C1(NC(C2CCCN2C(c2ccc(Cl)nc2F)=O)=O)CCCCC1(F)F N1(Cc2ccc(OC)nc2Cl)CCCC2(CC1)CNC(=O)O2 N1(C=O)CC2CCOCC2(NC(=O)CO)C1.C(=O)(CCC(C)C)c1c(OC)ccs1 C(=O)(CCS(N)(=O)=O)N1C(CN(C(C(CCN(C)C)N(C)C)=O)C)COCC1 CC1=C(C(=O)NCCC(C)(C)NC(C2CCC23CCC3)=O)CCO1 C1(O)(CC(=O)N(C)CC2N(C(CCc3nc(C)sc3)=O)CCC2)COC(C)(C)C1 C1(C(N2CC3CC3(CO)C2)=O)CC(c2cc(F)ccc2F)=NO1 CC1CCC(C)(C(=O)N(C)CC2CCCCN2C(C2CC(C)(C)CO2)=O)CC1 C1(C)(N(C)CCOC)CCCN(C(=NCC2CC(OC(F)F)C2(C)C)NCC(F)F)C1 Cc1nc(NCC2CN(C(c3cscn3)=O)CC2C(F)(F)F)ccc1[N+](=O)[O-] c1(CC)[nH]ccc1C(=O)NCC1CCN(C(=O)COCc2nc[nH]n2)C1 C1(SCC)CCN(C(=O)COc2sccc2C(=O)Nc2cccc(C)c2)CC1F C1(CNC(C(C)C2CC2)=O)CCCC12CC2.C1=CCNC(=O)C1 c1(NC(C)=O)ncc(C(=O)NCC2CC2NC(c2ccc(NC(C)=O)s2)=O)s1 N1(C(C2(CCOC)CC2)=O)CC(OC)CC(NC(C2CCC(C(N)=O)CC2)=O)C1 N1(C(c2cc(F)n[nH]2)=O)CCC2(COC(CNC(C3(O)CCC3)=O)C2)C1 C1(CC(N2CC(OC)(CNC(c3oncc3C)=O)C2)=O)OCCCC1(C)C CC1(C)C2CC(C(N3CC(O)(CNC(=O)C=CC=C(Cl)Cl)C3)=O)CC12 C(C)(CSC)(C(=O)NC1(c2noc(C)n2)CC1)NC(CC(=O)OCC)=O n1(CC)c(C)cc(C(N2CCN(C(c3csnn3)=O)CC2COC)=O)c1C CC12CC(C(=O)NC3(CNC(c4cc(C5CC5)ccc4Cl)=O)CC3)C3CC1C2C3 N12CCOC(C1)CC(=O)NCCC2=O.C(CC(C)C)C(N(CCC)C)=O C(=O)(CC(O)CCC)NCC1C(NC(c2c(CCC)occ2)=O)CCCC1 c1(C(N2CC(O)(CNC(CSCCC)=O)C2)=O)cc(Br)c(CC)s1 C12(C(=O)NC(CC)(CC)C(F)(F)F)CCCC1CN(C(=O)CNC(=O)NC)C2 Cc1cc(C(=O)NC2CC3(C2)CC3NC(c2cn(CCO)nc2C)=O)cc(O)n1 c1(NC(CN2CCN(C3C(=O)NCC3)CC2)=O)ccc2ccc(Cl)cc2n1 Cn1cc(C(=O)NC2CC(NC(C3(C)CCC(=O)C3)=O)C2)c(=N)[nH]1 C(C)(C)(CCC(=O)N(C)CC1CC(F)CN1C(=O)CC1CNC(=O)O1)N(C)C C1(C2CCN(C(c3ccc(N)cc3)=O)CC2)(NC(CCC(C)(C)C)=O)CC1 N1(C(C2C3CN(c4nc(C)cc(C)n4)CC32)=O)CCC2(CCNCC2)CC1 c1(OCCC)ccnc(C(=O)NCC2C=CCN2C(C2CC2c2ccccn2)=O)n1 c1(C(=O)NCC(CNC(Cc2n(C)ncc2Cl)=O)O)cc(N)c(F)cn1 c1(N(C)C)ccc(C(=O)NCC2CCCCN2C(=O)CCCCCBr)c(F)c1 N1(C(C2N(C(C(C)=CC=C)=O)C(C(C)C)CC2)=O)CC2(C=CCO2)C1 c1(C(=O)NC2CN(C(CC(=O)NCC)=O)CC(O)C2)n[nH]c2c1CC(C)OC2C Cc1cc2sc(C(N3CC(n4cc(C5CCCCN(C)C5)nn4)C3)=O)cc2s1 O=C(CCCCc1ccc(Cl)nc1)NNc1cccnc1Br C1(=O)CCC(=O)NCC2CCCC(C2)CN1.c1(CC)nnc(N(C)CCO)s1 C(c1cccc(F)c1Cl)=CC(=O)NCC1C(NC(C2CCN(C)CC2)=O)C1 CC1(C(=O)NCC(C)(C)C2CC2)CCCN(C(C2CCCCC2)=O)C1 c1(C(C(=O)NC2CCOC2)N(CCOC)C2CC2)ccc(OC)nc1C c1(C(N2CC(CCNC(CSc3n(C)cnn3)=O)C2)=O)cc2ccncc2s1 C1(CNC(N(C2CCOC2C)CCC)=O)CCC2(CCCO2)CC1 C=C(Cl)CC(N)C(=O)NC(C1(C)CCCC1)CCc1cccnc1 c1(C(N2C(CNC(COCCOC)=O)CCCC2)=O)cncc2cnccc12 c1(C(N2CC(CNC(c3ccccc3)=O)C3C2C3)=O)cn2c(Br)cccc2n1 c1(-c2nc(C(CC)OC)n(C34CC(C(=O)OC)(C3)C4)n2)ccc(OC(F)F)c(Cl)c1 c1(C(=O)NCC(CNC(c2ncn(C(C)C)c2)=O)(C)O)cccc(N(C)C)c1 c1(C(=O)OC)ccc(C(=O)NCC2CC2NC(=O)C=CC2CCCO2)nc1C c12cc(Br)c(F)cc1[nH]c(=O)[nH]2.C1(COCc2ccccc2)CCCCC1F c1(OC)nc(=NCC2(C(C)(C)C)CCN(C(=O)C(C)(F)F)C2)nc(OC)[nH]1 C1(C(C)CNC(c2nc[nH]c2C(N)=O)=O)CCN(C(=O)CC(O)CN(C)C)CC1 C1(C(c2nnnn2C(C)(C)C)CCCN2CCCC2=O)(OC)CCCC2(CC2)C1 c1(CCC(N2C(CNC(C(CC#C)C)=O)CCC2)=O)c[nH]c2ccc(C)cc12 CC(CN=C(NCCN1CCCCC1C)NC1CCC1)Oc1ccc(F)cc1 c1(C(=O)NCCC(C)NC(c2cc(CC)on2)=O)c[nH]c2c(Cl)cccc2c1=O C(=O)(C(Cc1ccccc1)C(C)N)C(=O)OC(C)(C)C.c1(CSC)cnn(C)c1 C12(C(N3CCN(CC#C)C(=O)C3)=O)CCCC1CN(C(C1CC(C)(F)C1)=O)C2 C1(C2CCN(C(=O)C(C)CN(C)C)CC2)(NC(c2c(C)cc(F)cc2)=O)CCC1 Cc1[nH]c(C)c(C(N2CCC(C(C)C(=O)NCC3CC(CN(C)C)C3)CC2)=O)c1C N1(C(CC2C=NN(C)C2=O)=O)CC(NC(C2CC(F)(F)C2)=O)CC(C)(C)C1 c1(OC)cc(CC(=O)N(C)CCN(C(=O)CC2CCCO2)C)cc(Cl)c1 c1(C(N2CCC(NC(C3CCCS3(=O)=O)=O)C2)=O)cc2ccc(Cl)c(F)c2o1 c1(OC)cccc2c1C(C(=O)N(C)CCN(C)CCNC(c1cncs1)=O)CC2 c1(NC(C2CC(F)CN(Cc3cccn3C3CC3)C2)=O)ccc2c(c1)CCC2 C1(C(=O)NC2CC(N(C(=O)CN3CCS(=O)CC3)C)C2)CCc2nn(C)cc2C1 n1(CC)ncc2c(N3CCCC(C)(NC(C45CCOC(C)(C4)C5)=O)C3)ncnc12 C(CNC(c1[nH]ccc1C)=O)(CC(=O)NCCC1CCCCCC1)OC c1(NC(CCn2c(C)ncc2)=O)cccc(CNC(=O)CSCCC(C)C)c1 CC(CNC(=O)C(C)(C)O)C(=O)NCc1nncs1 c1(CC(=O)N)ccc(SC)cc1.CCC(Cn1ccnc1)CC N1(C(C2CCC(OC)CC2)=O)CCN(C(C2CC(F)(F)CS2)=O)CC(C)C1 c1(NC(C(C2CN(N3CC(C4CC(F)(F)C4)C3)C2)OC)=O)ccccn1.C(=O)C C(=O)(C(COC)(CC)CC)NC1C=CC(C(=O)NC(C#C)CC2CC2)C1 C1(CC)(CO)CCCN(C(c2ccc(Cl)c(Br)c2)C(=O)NC(C)CC)C1 N1(C(C2(C)C=CCC2)=O)CCC(C(O)CC(=O)OC(C)(C)C)CC1 c1(C(=O)NCC2C(C)CCN2C(=O)CCC(C)(C)C)cc2ncc(Br)cn2n1 Cc1[nH]nc2ncc(C(=O)NC(C)C(C)NC(=O)C(F)(F)C3(O)CCCC3)cc12 c1(CCC(=O)N(CC(C)N(C(C=C(C)C)=O)C)C)cccc(F)c1 n1(CCC(C)C)cc(C(=O)NCC2CC2NC(=O)CCc2cscn2)nn1 Cc1cncc(C(=O)NCC(O)CN(C(=O)C(c2cccc(Cl)c2)O)C)c1C C12(NCc3c(C)noc3)CCC(C(=O)Nc3ccc(NC(N)=O)cc3)(CC1)CC2 c1(CC(N2CC(CC)N(C(=O)CN(C)C(C)C)CC2)=O)cccc(F)c1[N+](=O)[O-] C(C(CC(=O)N1CCC(CO)C1C)NC(=O)CCCn1ccnc1)OC C=CCCN=C(NCCN1CCC1)N1CCC2CCCCC2C1 C1(NC(c2ccn3ccnc3c2)=O)CCC2(CC1)CN(C(C1CC1Cl)=O)CCO2 c1(C(N2CCC(NC(C3C=C(C)CS3)=O)CC2C)=O)ccc2c(c1)SCC(=O)N2 c1(-c2c(OC)ccc(F)c2)cc2c(C(=O)Nc3ncco3)coc2cc1N c1(C(=O)OC)ccc(CNC2CCC(NC(c3sccc3C(C)=O)=O)C2)cn1 C(=O)(C1=CC2(CCN(C(=O)CC(C)n3cccn3)C2)C1)NC(C)C C1(CNC(c2c(C)ccc(C)n2)=O)CCCC2(CN(C(=O)C(C)C3CCC3)C2)O1 c1(CNC(C(n2cc(Cc3ccccc3)nn2)C)=O)ccc(-c2ncc[nH]2)cc1 c1(C(N2CC(CNC(COCCC)=O)CC(O)C2)=O)cc2cc(C)ccc2o1 N1(C(C(C)C(F)F)=O)CC(C)OC2(CCN(C(=O)CCc3cnco3)CC2)C1 c1(OC)ccnc(C(=O)NCCC2COCCN2C(=O)CC2(CO)CC2)c1OC N1(C(C(n2ncc(C)c2)C)=O)CC2CCN(Cc3ccccc3)CC12 c1(CC)c(Cl)nc[nH]c1=NCC(C)(CC(C)C)NC(C1CCC(CC)O1)=O c1(C(N(C2CCN(C(=O)Cc3ccsc3C)C2)CC)=O)cn(C)ccc1=O N1(C(C(c2n(C)nnc2)(F)F)=O)CCCC2(CCCCC2NC(C2CC2F)=O)C1 C1(COC)CN(C(c2ccncc2Cl)=O)CCN1C(=O)CC(F)(F)Br N1(C(=O)C(F)C2CC2)CCN(C(=O)Cc2c(Cl)cccc2Cl)C2CS(=O)(=O)CC12 c1(NC(C23CC2CN(Cc2c(F)cc(Cl)cc2F)C3)=O)ccc2ccccc2n1 C1(CC)C(NC(=O)CC2CSC2)CCCN1C(c1ccc(N)cc1F)=O CC1CCC(CNC(=O)CN(C(=O)Cn2cccn2)C2CCC2)C1 C1(NC(CCOC(C)=O)=O)CC2(C1)CC2C(=O)NCc1nccc(C)n1 C(C)(CO)(C(F)F)NC(C(C1CN(C(C(C)c2ccsc2)=O)C1)O)=O Cc1cc(C(=O)NCCOC2CN(C(=O)C(C3CCOCC3)C)C2)cnc1F C(=O)(C(C)(C)C(C)(C)O)NCc1nnn(C)c1C(N1CCC2(CC1)CC2CO)=O Cn1ccc2cccc(ON3CCC(S(CC(=O)N=c4cc(Cl)o[nH]4)(=O)=O)C3)c12 C1(NC(c2nccc(OC)c2)=O)CCCC12CN(C(C1CNC(=O)N1)=O)C2 Cn1c(C(=O)NCC23CC2CN(C(c2csc(-c4ccco4)n2)=O)C3)cnc1O C(=O)(CC1COc2ccccc21)NC(CC1CCN(C(C=C(C)Cl)=O)CC1)C c1(C(=O)NC(C)CN(C)C)cc(CNC(C2CCSC2)=O)nn1C c1(CC(=O)NC(CC)CNC(C2(CC)CCC(O)CC2)=O)cn2ccccc2n1 C1(C(N2CCC(C3CC3)C2C(=O)NCCC2CC2)=O)CCn2cnnc2C1.C1CC1 CC1CC(C(=O)COC(F)F)CC(C)C1.C12CCCN(C1)C2c1ccccc1 N1(C(c2c(NC)nsn2)=O)CCC2(CCCC2C(N2CCC2C(=O)OC)=O)C1 c1(NC2CCN(c3cc(C)[nH]n3)C2)nccc(=NC(CCO)c2cccc(Cl)c2)[nH]1 C1(NC(=O)CN2CC3CC3C2)CN(C(=O)C=C2CCCC2)CC1C1CC1 C(=O)(CCC(=O)c1ccc[nH]1)N1C(CNC(=O)Cc2ccc(C(N)=O)nc2)CC1 C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1C(NC(C2(SC)CC2)=O)C1 c1(C(N(C)CC2(NC(C3CCC(C)(C)C3)=O)CC2)=O)cc2cccnn2c1 C(C(F)C(=O)OC(C)(C)C)N(CCNC)C(C1(NC(C)=O)CC1)=O.C1(SC)CC1 C(=O)(C(C)CC(F)F)NCC(CO)NC(c1n(CC)ncc1Cl)=O n1(CC(=O)NCC(C)CN(C)C(C2CCOC2=O)=O)ncn2nccc2c1=O Cc1c2c(nn1C)CC(NCc1cnncc1C(F)(F)F)CC2 C1(CNC(=O)CC2CCC3CC23)CCCC1NC(=O)CNC(=O)CC1CCCC1 n1(C(C)C(=O)NCC(C)(C)CC2CN(C(C3(CCO)CC3)=O)C2)cc(Cl)cn1 N1(C(CCNC(=O)NC)=O)C2CC1CN(C(=O)Cc1cnco1)C2 c1(C(N(CCNC(CCN(CCC(C)(C)C)C)=O)C)=O)c[nH]ccc1=N N#CCC(C(F)(F)F)OC(C1CC2C=CC1CC2)=O Cc1ccc(C(=O)NCC2CCCC2NC(c2c(Cl)n[nH]c2C)=O)c(N)c1 C1(C(=O)Nc2ccc(CCF)cc2)CC2CC1CN(C(=O)C=Cc1ccco1)C2 c1(C(=O)NCCN(C)Cc2ccccc2Br)cc(=O)n2ccsc2n1 CC1CN(C(=O)CN(c2ccccc2)C)CC1CCN(C(=O)CC1CCCO1)CC C1(NC(c2ncc(N(C)C)nc2)=O)CC2CC(NC(c3cc(F)n(C)n3)=O)CC12 C1(CNC(=O)C(F)C(F)(F)F)CC2(CO1)CN(C(c1ccn3nnnc3c1)=O)C2 c1(NC(=O)NC(c2ccncc2Cl)C)ccc(N2CCNC2=O)cc1 c1(NC(C(=O)NCC=CC(=O)Nc2nc(OCC)sn2)=O)ccc(N)cc1 c1(-c2nc(C3(C(F)(F)F)CCCO3)on2)ccc(C)cn1 c1(C(N2C(C)CC(NC(c3csc(O)n3)=O)C2)=O)cc2c(cc1F)NCCC2 C(=O)(CCCC(F)(F)CO)Nc1ccc(NC(C(C(=O)OC)C)=O)cc1C C1(C(=O)OC)CN(N2CCC3(CCNC3=O)CC2)C(C)(C)CO1 c1(C(N2CC(NC(C34COC(C3)C4)=O)C2)=O)cnc(-c2ccccc2)nc1 c1(C(=O)Nc2c(Cl)ccc(OC)c2)ccc2c(c1)CN(Cc1ccc(=O)oc1)C2 Cc1ncc(CN(C2CCC(c3nn[nH]n3)O2)C)[nH]1 c1(OC)cc(Br)c(Cl)cc1C(N1CCN(C(C#N)C(C)C)CC1)=O c1(CC)cc(C(=O)N(CC)CC2CCCN2C(c2sccc2OC)=O)n[nH]1 N#Cc1ccc(OCC(N2CCC(=CCNC(=O)CCF)CC2)=O)c(Br)c1 C1(NC(C2OCCN(C(C3(C=C)CCOCC3)=O)CC2)=O)CCC(=O)NC1(C)C C1(C(=O)NC(C)CNC(c2csc(-c3ccccn3)n2)=O)CCCS(=O)(=O)N1 Cc1cc(C(=O)N(CCCNC(=O)C=Cc2cncc(O)c2)C)nc(C)n1 C(=O)(C(C)(C)CCC(=O)OC)N1CCC(C2CC2)(NC(C(CC)OC)=O)C1 C1(C(N2CC(O)(CNC(c3cc(CCC)nn3C)=O)C2)=O)CCn2cncc2C1 CC(C)(C#Cc1cn(Cc2ccc(Br)cn2)nn1)OC.S(C)(=O)(=O)CNC(=O)CN c1(C(=O)OC)ccc([N+](=O)[O-])c(NCCOCCNC(=O)C(C)OC)n1 CCC(CC(C)C)C(=O)N1CC(NC(=O)Cc2ccc(O)c(Cl)c2)CC(F)C1 CC(C(=O)NC(CNC(=O)CC1CCCNC1=O)CO)C1=CCCC1 N1(C(Cc2c(C)nccc2)=O)CCC2(NC(c3cnn(C)n3)=O)CCCCCC12 CC(C)C(C)C(=O)N1CCC1CNC(C1(C(C)(F)F)CCC1)=O c1(Cn2cc(-c3cccc(C(C)C)c3)nn2)cc2ccccc2n1C N1(C(c2ccc(C(C)=O)[nH]2)=O)CCC(CNC(C2CC2C)=O)C(C)C1 C12(C(N3CCC(CNC(C4C(C)OCC4)=O)(CO)CC3)=O)CCC(CC1)C(C)O2 c1(CCC(=O)NC2CC2CNC(C2(Cl)CC2)=O)ccc(Cl)s1 C(CC(C(=O)N(C)CCn1ccnn1)NC(=O)CC(CC)SC)=CC N1(C(C2(CN(C)C)CC2)=O)CC2OCCN(C(c3cnc4c(c3)NCC4)=O)C2C1 C(=O)(C(CC)C(C)O)NC(CNC(C1(CC#C)CCCC1)=O)(C)Cn1cccn1 N1(C(C=Cc2ccc(C)s2)=O)CCCC(NC(=O)C(C2CCCCC2)N(C)C)C1C CC(C)(C)CCCCC(=O)NCC1CC(NC(C2CCOCC2(C)C)=O)C1 O=C(CC1=CCC(C(=O)Nc2ccc(C3CCO3)cc2)CC1)N1CCCC1 c1(C(=O)NCC2(C)N=C(C)SC2)cnc(Cl)c(C)c1 Cc1cc(S(N)(=O)=O)cc(C(=O)NCC=CCNC(=O)CCc2csc(=N)[nH]2)c1C N1(C(c2n[nH]c(C)c2O)=O)CC(C)(C)OCC1CNC(=O)C(O)CC(C)C N1(C(c2nn(C)c(Cl)c2)=O)CC(NC(C2CCCCC2C(N)=O)=O)CC12CCC2 c1(C(=O)NC2(CC=C)CCCC2)cncc(CNC(=O)C=CC(=O)OC(C)(C)C)c1 C(=O)(C(C)(C)CCCC(=O)N(CC(C)CNC(C1CC(C2CCC2)C1)=O)C)OC N1(C(C(CCC)O)=O)CCN(C(=O)CCc2ccc(O)cc2)C(CO)C1 NC1CC2CC2C1.C(=O)CCCC1CCCS1 c1(OC)ccc(Br)c(C(C)NC(C2CCCC2)C)c1F c1(C(c2nnnn2CCOCSc2ccc(OC)c(Cl)c2)OC)cccc(C)c1Br N1(C(CCCCC=C)=O)CCC(NC(c2ccnn2CC#N)=O)C(F)(F)CC1 CC(C)S(=O)(=O)C(C)C(=O)NCCN(C(c1cc2cccnc2s1)=O)C1CC1 N1(C(C2C(C)C2)=O)CC(NC(c2cccc(CO)n2)=O)CC12CCCOC2 c1(NC(=O)C(Cl)(Cl)Cl)ccc(NC(C2CCCC3CC23)=O)cn1 C(=O)(C1=COCCC1)N(C(C)CCNC(=O)CCC1CC1(C)C)C C(=O)(C1=CCC2CCC1N2C(C1C2CCCC12)=O)NC1(C)CCC(C)C1 c1(C(N(C)CC2(O)CCN(C(C(C)OC)=O)C2)=O)c(C)nn2cc(C)cnc12 S(=O)(=O)(c1cnc(NNS(C)(=O)=O)c(Cl)c1)NCC(C1CCCC1)O N1(C(C2C(C)CCS2)=O)CC2CC(C1)CN(C(=O)CC(C)(C)CN(C)C)C2 N1(C(C(CC)C2CCOCC2)=O)CC2CN(C(=O)C(c3cccn3C)=O)CCC12 N1(C(CC(=O)OC)=O)Cc2nccn2CC(NC(c2ccc(C(C)C)cn2)=O)C1 N1(C(C2=CCCC2C)=O)CCN(C(=O)Cc2cccnc2)C2COCC12 c1(C(=O)NC2CC3(CN(C(C(C)OCC)=O)C3)C2)ccc(Cl)c(Cl)c1O C1(CC)CCN(C(=O)CCC2CCCC2)C1C(=O)Nc1cn(C)nc1C(C)C N1(CCOCC=C)CCC2(CN(C(c3scnc3COC)=O)CC(C)O2)C1 C1(C(=O)NC2(CCC(=O)NC(CC)C(=O)OC)CCC2)CCC(O)CN1C c1(C(C)C)nocc1C(N1CCC(N2CCCC2=O)C1)N(C)C c1(CC)cccnc1C(N1CC(O)(C(F)C(=O)NCC(=O)NC(C)(C)C)C1)=O C(=O)(C(CNC(=O)CSC(C)(C)C)C(C)(C)C)N1C(C=C)CC1 C(c1ccc2c(c1)OC(F)(F)O2)=CC(=O)NCC(CN(C(C(CC)(F)F)=O)C)O [N-]=[N+]=NCCCCCCC(=O)N1CC(CNC(=O)C(C2CCOCC2)F)C1 Cc1cccc(NC(=O)C(C)(C)C2CCCN2C(=O)CSc2ccccc2C)c1 N1(C(c2ccc(CC)o2)=O)CCC2(CC1)CC2CNC(C1(C(F)(F)F)COC1)=O N1(C(CC=C(C)C)=O)CCN(C(=O)C(=Cc2ccccc2)OC)CC1C1CCC1 C(c1cccc(CO)c1)=CC(=O)N(C1CCCN(C(=O)Cc2cncs2)C1)CCO N1(C(=O)CCc2ccc(Cl)c(Cl)c2)CC(C2CN(C(C3CCC(F)C3)=O)C2)C1 N1(C(C2(CCCC)CC2)=O)CC(F)(CNC(c2ccc(-c3csc(C)n3)s2)=O)C1 C1(NC(c2cnsn2)=O)CC(O)CN(C(c2cn[nH]c2)=O)C1 C1(NC(C2C(C)C2)=O)CCC(N(C)C(c2cnc(Cc3ccccc3)s2)=O)CC1 C1(COC)(NC(c2cncc(Br)c2)=O)CCN(C(C2CC2C#N)=O)C1 C#Cc1ccc(OC)c(C(=O)NCC2CCN2C(c2cnc(COC)o2)=O)c1 C1(NC(C2(C#C)CCC2)=O)CCN(C(c2cc(OC)ns2)=O)C1C(C)(C)C C1(NC(C2N(C(C)=O)CCOC2)=O)CN(C(=O)CC2CC(C)(C)C2)C(C)(C)C1 C(C)(CC(=O)N1CC(C(O)C(=O)NC2CC(N(C)C)C2)C1)SC C1(C(N2CCC(F)(CF)C2)=O)CCCCN1C(=O)CC1(CO)CCC1 N1(Cc2cnc(C(=O)O)s2)CC2C(C1)N2C(c1cccnc1Cl)=O C=CC(C)(C)C(=O)N1C(C(=O)NCC2CCC(F)C2)CC2CC12 c1(C(N2CC(C)(NC(C3N(C(C)C)CCC3)=O)C2)=O)ccc(O)c(C(C)(C)C)c1 C1(C(=O)NCC(C)NC(=O)C(O)CC2CCCC2)CCC(C)(C)O1 c1(-c2cn(CC)nn2)ncc2ccccn12.c12onc(C(F)(F)F)c1C(=O)NC2 S(=O)(=O)(c1ncccc1Br)N(C(Cc1ccccc1)C(=O)O)CC(=O)NCCO Cn1nc(C(=O)NC2(C(N3CCC(CCO)C3)=O)CC(F)C2)cc1O N1(C(c2cc(C)no2)=O)CC2CCN(C(=O)CCc3cccnc3)CC12 C1(CC(=O)NCC=CCNC(=O)CCSC(F)(F)F)(C(=O)NCC=C)CCCC1 Cc1cc(Cl)ccc1CC(N1CCCC(O)(CNC(=O)C(C)CCN(C)C)C1)=O C1(C(=O)NCCOC)CNC(=O)CN1C(=O)C(C)S(C)(=O)=O C1(C(N2C(C)(CNC(C(C(C)C)n3cncn3)=O)CCC2)=O)OCCN(C)C1=O CC1CN(C(=O)OC(C)(C)C)CC1C(C1CCC1)NC1(c2cccs2)CC1C CCCCC(O)C(=O)N1CCC(C)C1C(N1CC(C2CC2)(CC)C1)=O C(=O)(C1=CCCC1)N(C1CC1)CC1N(C(C(Cn2ccc(C)n2)C)=O)CCC1 c1(CC)nc(O)sc1S(=O)(=O)NC(c1ccc(C)cc1Cl)CCO S(=O)(=O)(c1ccccc1Cl)NCC(N1C(CNC(C(C=CCCC)O)=O)CC1)=O c1(C(N2C(C(N3CC(CC(C)C)OCC3)=O)COCC2)=O)c[nH]c2cnccc12 c1(C(N2CC(C(C)NC(c3cc(C)ncn3)=O)OCC2)=O)cc(O)nc(O)c1 C1(NC(Cc2nc(=N)[nH][nH]2)=O)CC12CCC(NC(C13CC(F)(C1)C3)=O)CC2 CC(O)(CC(F)(F)F)C(=O)N1CC(C(=O)NCCN2CCN(C(=O)C(N)=O)CC2)C1 c1(CC)cncc(C(=O)NCC(C(=O)NCCC(C)C)N(C)C)c1 C1(OC)CC2(C1)CC2N=c1[nH]nco1.n12nccc1C(=O)NCC(=O)N1CC2C1 CC1(C)CCN(c2nnc(COC(F)F)n2Cc2ccccc2N2CCC2)CC1 O=C(CNC(N1CCN(c2ccc(C(F)F)cc2)CC1)=O)NNc1ccccn1 CC12CC(CS(=O)(=O)NCc3nc(Cc4c(Br)ccn4C)no3)(CO1)C2 N1(C(c2cnc3sc(C)c(C)n32)=O)CCCC2(C1)CN(C(=O)C(C)C#N)CCO2 C12(C(N(CCNC(c3cc(C(F)(F)F)no3)=O)CC)=O)CC3CC1C2C3O N1(C(C(C)n2cnnn2)=O)CCC(NC(c2cccc(C(F)F)n2)=O)CC(O)C1 c1(C(=O)NC2CC(CNC(C3C(OCC)C3C)=O)C2)cc(N)cnc1Cl Cn1ccnc1C(C)(C(=O)NCCCOCC1CCCO1)O.N(CCO)(C1CC1)CC1CC1 Cc1cc(C(N2CCCC(CN(C(=O)CC3NC(=O)NC3=O)C)C2)=O)cc(Cl)c1 C1(CC)CCCC(N=c2[nH]c(N3CC4(CCCO4)C3)nc3ccsc23)C1 N1(C(CCOCCC)=O)CCN(C(c2cc(C3CC3)nn2C)=O)C(C)C1C CC(C)CC(C(=O)NCC1CC(NC(=O)CC2CCC2(F)F)C1)NC(N)=O N1(C(c2cccc(OCCC)c2)=O)CCC(C)C(NC(=O)C(F)=C2CCC2)C1 C12CCC(CC1)C(=O)N2C1CC1.N(C(=N)N)CC c1(C(=O)OCc2c(OC)c(F)ccc2)cc(S(=O)(=O)Cc2cccnc2)ccc1F CC(C)C(C(=O)OC(C)(C)C)C(=O)NCCC(O)CNC(C1(Cl)CC1)=O Cc1cc(Cl)cc(C)c1C(=O)NCC12CCC1CCN2C(c1nc(=O)n(C)[nH]1)=O CC1OC2(C)CC1(C(N1CCC(NC(=O)CCC(F)(F)F)C1(C)C)=O)C2 c1(NC(C=C)=O)ccccc1-c1cc(C(N2CCOCC2C)=O)ccn1 C1(C(=O)NCCCC2N(C)CCC2)CCCN1NC(=O)CCC1CC1 C1(C(N(CC)CC)=O)CN(C(c2ccc(-n3cccc3)cc2)=O)CCC1O C1(C(=O)Nc2ncccc2I)CN(C(c2cc(Br)ccn2)=O)CCC1O CCCC(C(=O)NC1CC(NC(=O)C(C)Oc2cccc(OC)c2)C1)N(C)C N1(C(C2N(CCC)CCC2)=O)CC2CC1C2CNC(c1cc(Cl)no1)=O N1(C(c2cnc(CC)nc2)=O)CCC(C(=O)NCC2CCC2(F)F)C1(C)C c1(C(=O)NC(CN(C(=O)Cc2cccs2)CC)C)cn(C(F)(F)CO)nn1 CC(C)CC(CNC(C1(C(C)F)CC=CC1)=O)NC(=O)C(C)Cc1ccccn1 c1(C(N2CCCCC(N(C)C(c3cccc(Cl)c3)=O)C2)=O)ccccc1S(C)=O c1(NC(=O)NCCCc2ncc(OC)nc2)c(F)cc(Cl)cc1Br c1(CCCC(=O)NCCOCCCNC(C2C(C(N)=O)CC2)=O)ccccc1Cl c1(C(C)C)nc(N(CCC#N)C)cc(N2CCN(c3cn[nH]c3)C(=O)C2)n1 c1(-n2ncc(C(=O)NC3(CNC(C4CCC(=O)C4)=O)CCC3)n2)cccc(Cl)c1 O=C1Cc2cc(C(N3CC4CC3CNC4)=O)ccc2N1.N12CCC(CC1)C2 C1(C(C)NC(C2(F)CC2)=O)CCN(C(=O)CCC2CCCC(O)C2)CC1 C1(NC(=O)C2=CCCS2)C2CC(O)C1N(C(c1cncc3ccsc13)=O)C2 c1(C(N2CCN(C(c3ccncn3)=O)C(CF)C2)=O)ccc(F)c(Cl)c1 c1(CC)n[nH]cc1C(=O)NC1(C)CC(NC(C2CN(CC(C)C)C2)=O)C1 C1(c2cn(CC(Cl)CO)nn2)(COC)CCSCC1 C1(C(N2CC(N(C(c3n(CCOC)ncc3)=O)C)C2)=O)C2CC3C(C2)C13 c1(C(c2onc(-c3cc(C)ns3)n2)(F)F)ccc2c(c1)OCCCO2 Cc1ccc(C(N)=O)cc1C(N1CC(CCNC(=O)C2=CCCS2)C(C)C1)=O N1(C(C(c2ccncc2Br)C)=O)CC2CCC1CN2C(c1cnsc1)=O C(=O)(C(C)(C)CC(C)C)NCC(CNC(c1cccc(CCC)c1)=O)F C1(C(N2C(CC(=O)N(C(c3ncccn3)C)C)CC(O)C2)=O)C2CCC(C2)C1C N1(C(C2(CC)CCOCC2)=O)CCC(NC(c2oc(C)cc2C)=O)C(O)C1 C(=O)(C1Cc2ccccc21)NC1C(C(=O)Nc2ccc(OCC)cn2)C1(C)C.OCC N1(C(C(CCC)C)=O)CC(NC(=O)CN2C(=O)CN(C)C2=O)C(C)(C)C1 CC1CCN(C(=O)C(c2ccc(F)cc2)(C)O)CC1NC(C1(CO)CCCO1)=O C1(CNC(C2(OC)CCSC2)=O)CN(C(=O)C(F)(F)C(O)C2CC2)CCC1(C)C c1(-c2nc(CC(CC)C)nn2CC(C)C2CC2)ccc(F)c2occc12 C1(NC(=O)COc2cccnc2)CN(C(=O)C=Cc2ccc(F)cc2)CCC1F n1(CC)nc(C)c(CC(=O)N(C2CCS(=N)(=O)C2)C)c1C.c1(C)ccccc1Cl C1(C(=O)NCC(C2CCCC2)NC(CSCCC)=O)CCC(C)C1 C(CC(C)C)(C(=O)NCCc1cc(C)[nH]n1)NC(c1cc(CC)sn1)=O Cc1cccc2c1OCCC2NC(N1CC(c2ccoc2)CC1C)=O c1(OCc2nnc(N(CC=C)CC=C)n2Cc2cccs2)ccc(C)cc1C C1(CNC(COCCOC)=O)CCCC2CN(C(=O)C(C(C)C)N(C)C)CC12 c1(C(=O)NC2C3CN(C(C(CC)(F)F)=O)CC32)cc2c(s1)CCSC2 CC(CN(C)C)CCC(=O)N1CCN(CC(=O)NC(c2cncnc2)C)CC1 N1(C(C=CC)=O)C2CCC1CC(CC(C)NC(C1CCCCC1(F)F)=O)C2 c1(C(=O)NC(c2cn(-c3ccc(Cl)cc3F)nn2)C)cnn2cccnc12 c1(C(C)=O)ccc(C(=O)N(C)CC2CCCN2C(C2(C)CCNC2=O)=O)cc1F C1(NC(C2(c3ccccc3)CC2)=O)CC2CC(NC(C3C4COCC34)=O)C1C2 Cc1cnc2cccc(C(=O)NCC3CCN3C(c3[nH]c(=N)sc3C(=O)O)=O)n12 C(=O)(CCCCCN=[N+]=[N-])N(CC(C)CNC(c1nccc2cc[nH]c12)=O)C C(N=c1[nH]c(N(C)Cc2ccnn2C)nc2c1CCCC2)c1cc(OC)nn1C c1(OC)ccc(C(N2CCOCC2CNC(=O)C(C)CSC(F)(F)F)=O)c(O)c1 C1(n2ncc(C)c2)=CC(NCc2ccc(N3CCN(C)CC3)nc2)=NC=NO1 N1(C(CCSC)=O)CCC(C2CCCN(C(c3nocc3Br)=O)C2)C1 CC1=NOC(C)(C(=O)N(C2CCN(C(C3(Br)CC3)=O)CC2)CC2CC2)C1 C(=O)(CC(C(C)(C)C)NC(c1csnc1C)=O)NC1CN(CC)CC1C c1(CC(=O)NC2(CO)CN(C(Cc3n(C)ccn3)=O)C2)ccc(Br)c(O)c1 N1(C(C(C(=O)OCC)OC)=O)CC(CNC(c2ccc(F)s2)=O)C2(CC2)C1 C1(C(N2CCC(NC(C(C(C)C)=O)=O)(CF)C2)=O)CCC(O)CN1C C1(NC(C(C)OCCCC)=O)CCCCN(C(=O)CC2CCCO2)CC1.C(C)(=O)O N1(C(Cc2nc(C)sc2)=O)CCN(C(=O)C=CC2CCC2)CC(C)(C)C1 c1(OC(C)C)ccc2oc(=O)c(C(N3CCC3C3CCC3)=O)cc2c1 C=C(C)C(C)(O)CNC(=O)C(=O)NC1CCOC(C(C)C)C1 c1(C(N2CCC(O)(CN(C(c3c(C)scn3)=O)C)C2)=O)cccc2c1OCC2C CC(C)C(C(=O)NCCN(C(c1cnc(S)nc1)=O)C1CC1)N1CCCS1(=O)=O c1(N)cc(C)cc(C)c1.c1(C(N(CC#C)CC)=O)csc(CNC(C2CCOC2)=O)c1 C1(NC(CC=C(C)C)=O)(CNC(=O)C(c2ccc(C)o2)C)CC2CCC1CC2 C(=O)(CCC(C)O)N(CCNC(CC1ON=C(C)C1)=O)C(C)C c1(OC)cc(OC)c(NC(C2CCCCC2C)=O)c(OC)c1 Cc1nn(C(C)(C)C)c(C(c2nnnn2C)NC2CCCN(C)C2)c1Br c1(C(=O)NCC(CNC(C2CCCOC2)=O)OC)ccc2nnc(C)n2c1 C1(C(=O)NCC(C(=O)OCC)C)(CF)CCN(C(=O)CN2CCCC2=O)C1 C(C)(CNC(C1CCC(C)(C)CC1)=O)(CC(C)C)NC(CN1CCC(OC)C1)=O c1cc(F)ccc1C.c1(C(N2CCCC2(c2ccccc2)C)C)ccccc1F c1(NCCCOC)ccc(-c2ccc(C(=O)N=c3ccs[nH]3)cc2)cc1[N+](=O)[O-] C(C)(N=c1cc(C)nc(N2CCn3nc(C)cc3C2)[nH]1)c1ccc(OC)cn1 N1(C(C=C(C)Cl)=O)CC2CC3CC2C1C3NC(c1n[nH]c(C)c1C)=O c1(OC)ccc(Br)c(NC(C2CC2C(=O)N(C)CCc2ccccc2)=O)n1 N1(C(CCN(C)CC)=O)CCCC(NC(=O)CCc2cccc(F)c2F)C(F)C1 C(=O)(CC(O)CCSC)N1C(CNC(CC2(OC)CC2)=O)CCCC1 C1(NC(C=C(C)C)=O)CC2CCC1N2C(C1CC1[N+](=O)[O-])=O C1(CNC(c2ccc(C(C)=O)[nH]2)=O)CCN(C(C2CCCC2O)=O)C(C)C1 Cc1ccc(C)c(C(N2CCC(NC(C3CC4(C3)CC4F)=O)C23CC3)=O)n1 c1(NC(C(C)OC(CC(CC)O)=O)=O)ccc(C=CC(F)(F)F)c([N+](=O)[O-])c1 N1(C(c2ccc(CC)[nH]2)=O)CCC(C(F)(F)F)C(CNC(=O)Cc2nc[nH]n2)C1 Cc1nc2ccc(CNC(C34CC3CN(c3ccnc(C(C)(C)C)n3)C4)=O)cc2o1 CC(C(=O)NC1(C(C)O)CC1)NC(=O)CCc1cncs1 CC1=C(C(=O)NCC(C2CCCN2C(=O)CN2CCCS2(=O)=O)(C)C)SCCO1 C1(NC(=O)COCC2CC2)CCC(NC(=O)CCCc2cncs2)CC1 C(=O)(C(CNC(C1COCC(C)O1)=O)C(C)C)NC(CCOC)C Cc1cnn(C)c1C(=O)NC1CCN(C(=O)C(C(C)C)n2cncn2)C1C1CC1 N1(C(CCC(=C)Cl)=O)CCC(C2CCN(C(=O)CCCc3n[nH]c(=N)s3)C2)C1 C(=O)(CC(C)CCC)NC1(CC=C)CN(C(c2cn(C)cc2C)=O)C1 c1(C(=O)NC(C2(O)CN(C(C(N3CC(C)C3)C)=O)C2)C)nn2cccnc2c1Cl C1(C(=O)NCc2cn(CC(=O)NC(C)CC(C)Cl)nn2)CCCOC1C C1(OC)CCC(N=c2[nH]c(N(C)CCc3ccccc3Cl)nc3c2CCC3)C1 c1(OC)ccc(C(=O)NC(C)CNC(C2CC(=C(F)F)C2)=O)c(OC)n1 C1(C)(C(=O)OCC)CCN(C(C2C=CCC2)=O)C1.C12CCOC1NC2=O S(=O)(=O)(c1ccc(F)cc1)N1C2CC(NC(C(CCC)Cl)=O)CC1CC2 c1(OC(c2onc(COCC)n2)=O)ccccc1F C(C)(CC(C)NC(c1csc(-c2cccs2)n1)=O)NC(CC=CC=C)=O CCCCCCC(C)C(=O)NCCCNC(=O)Cc1cnsc1 C(CO)(CCCCN(C(c1cc(-c2ccc(F)cc2)[nH]n1)=O)CC)NC(C=CC)=O C(C(CO)C(F)(F)F)NC1c2conc21.c1(C(C)(C)C)nnnn1CCCF c1(CC)nn(C)c(CC)c1C(N1CC=C(CNC(=O)Cc2ccn(C)n2)CC1)=O c1(C(C(=O)N(C2CC(O)C2)C)NC(CCOCC#C)=O)ccccc1 C1(C(N2CCC(NCc3ccccc3)CC2)=O)CCCN(c2ncccn2)C1 N1(C(C2(C)C(CC)CCC2)=O)CCC(=CCNC(=O)CCC2CCCN2C)CC1 C1(F)(CNC(C(CC)=CC)=O)CCCN(C(c2ccc(OCC(N)=O)cc2)=O)C1 C(=O)(C1CCCn2cc(C(C)(C)C)nc21)Nc1nn(C)c2c1c(C(F)(F)F)ccc2 C1(C(N(CC(CC)OC)C)=O)CC2(CCN1C(C1COCC(C)O1)=O)CC2 c1(C(N2CC3C(CNC(=O)Cc4ccon4)(C3)C2)=O)cc(Cl)nc2n[nH]cc12 C1(C(=O)NC(C)C(C)(C)CN(C)C)CCCCCC1NC(C12CCCCC1C2)=O c1(C(N2CC(OC)(CNC(c3csc(C)n3)=O)C2)=O)cnc(P(C)(C)=O)cn1 C1(CNC(=O)C=Cc2ncc[nH]2)CCCC(C(=O)NC2(CF)CCC2)C1 C(c1cncc(O)c1)=CC(=O)NC1(CNC(=O)C=Cc2cocn2)CCCC1 C1(CCC)CN(C(=O)Cc2cn(C)nn2)CCN1C(=O)COCC(=O)OC N1(C(C(CC=C)C)=O)CC2CCC1C1CN(c3nccn4nnnc34)CC21 c1(C(C)C)ccc(C(=O)NC2CCCN(Cc3ccccc3F)C2)cc1Cl c1(CNc2cn(C3CN(C(CCCCC(C)O)=O)C3)nn2)ccc2n[nH]cc2c1 C1(C(=O)NC2CC(C(N(C)CC3C(C)C3)=O)C2)CCC2(CCC2)O1 C(=O)(CCC(F)(F)F)NC(c1ccc(C(C)C)cc1)CNC(C1CC2CCC1C2)=O C1(C(=O)NCC2CCC2CO)C(C2CC2)CCN1C(=O)CC(F)(F)F C(CNC(C1(C)CC(F)(F)C1)=O)(C(C)(C)C)NC(C(C)OCc1ccccc1)=O c1(C(=O)NC2C(CNC(CCCC(N)=O)=O)C2)cc2n(c1)CCCNC2=O C1(OCC)CC2CN(C(=O)C(C)N(C(=O)COC3CC3)C(C)C)CC12 C12(C(=O)NCC(C)O)COC(C1)C(NC(C1CCC(C)(C)CC1)=O)C2 n1(CC(N2CCCCCC(NC(C(C=C)O)=O)C2)=O)ccc2ccc(F)cc12 C1(C(=O)NCCN(C(c2ccc(C(C)C)o2)=O)C2CC2)Cc2c(F)cccc2O1 N1(C(C(CCC=C)NC(=O)CC(C(C)CC)SC)=O)CCN2CCCCC2C1 C1(C2CCCN(C(=O)C(CCc3ccccc3)CC(C)C)C2)(C(=O)OCC)CC1 C(C(C)(CC)NC(C1CC=CCO1)=O)NC(CNC(=O)OC)=O Cc1[nH]nc2ncc(C(=O)NCC3(C)CCN(C(=O)C(F)C(C)(C)O)CC3)cc12 C1(NC(C2(NC(C(CCCOC)C)=O)CC2)=O)(CO)CC2CCCC12 N(C(=NCC1CCCC(C(N)=O)C1)NCC1(Cl)CCC1)C(C#N)CC1CCC1 c1(C2(C)C(C(N3CC(C)(NC(c4c(C)n[nH]c4C)=O)C3)=O)C2)ccc(F)c(F)c1 C1(O)(N(C(CCOCC=C)=O)C)CCN(C(=O)Cc2ccccc2C(=O)OC)CC1 C(C)(c1ccccc1C)=CC(=O)NCc1scc(C(=O)NCC2C(COC)C2)c1 Cc1cccc(C2CC(NC(=O)Cc3ccccc3CC3CC3)C2)c1 Cc1cccc(CNC(=O)CC2CCCN(C(C34CCC(CC3)CO4)=O)C2)c1F C#CC1CN(C(c2cc(C)c(F)cc2N)=O)CCN1C(c1coc(CC)n1)=O CCCC(CCCNC(=O)CN1CCCCC1)NC(C1(n2cnnn2)CC1)=O Cc1c(C(N2CCCCC2CN(C(=O)Cc2cncc(F)c2)C)=O)cncc1Cl C12(C(=O)NCC3(NC(Cc4n(C(C)C)ncc4)=O)CCC3)CCC(CO)(CO1)C2 C1(CNC(C2(C#C)CCC2)=O)CN(C(=O)CCc2c(C)ncnc2O)CCN1C c1(C(=O)NC(CC)Cn2ccnc2)ccc(-n2cc(CN(C)CC)nn2)cc1F c1(NC(=O)CC2CN(C(C3CCC(F)(F)C3)=O)CCO2)cccc(Cl)c1[N+](=O)[O-] C(=O)(CC(O)C(N)=O)N1CCN(C2C(COC)CCC2)CC1 c1(COC)ccsc1C(=O)NCC1(NC(=O)CC2(N3CCCC3)COC2)CCC1 CN1N=C(C(=O)N2C3CC2CN(Cc2ccc4c(c2)CCO4)C3)CCC1=O C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC(CC)CN(C(=O)C(F)OC)CC C1(NC(c2nc(COC)oc2)=O)CC(CNC(=O)CCn2cccn2)C(O)C1 C1(NC(=O)C=Cc2ccc(O)cc2)CN(C(c2ccc[n+]([O-])c2)=O)CCC1(F)F.N CC(C)(F)C(=O)N=c1ccn(CC2CCCN2)[nH]1 c1(SCC(=O)NCCC2CC(C(=O)NC3CC3C(F)(F)F)C2)ccc(Cl)cc1 Cc1cc(CNC(=O)CC2CN(C(c3ccc(CO)cn3)=O)CCO2)cc(O)n1 N#CCCCCC(=O)N1CCCCC1CNC(=O)CCCCCN1CCSSC1 C1(Nc2snc(C(=O)NC)c2C)CCN(C(=O)C(C)NC(C)=O)O1 C(=O)(C(CC(F)F)C1CCC1)NC1(CNC(C2(C)COC2)=O)CCCC1 C(C(C(C)(C)C)NC(=O)CCOC1CCC1)NC(C1(C)CCCS1)=O C(=O)(C1=CC2CCC(C1)C2)N(C(C)(C)CC(=O)NC1CN2CCC1CC2)C S(=O)(=O)(C1CCC2CCC1OC2)NCCc1ccc(OC)nc1 C1(NC(c2cccc(-n3ccnc3)c2)=O)C2CC(O)C1N(C(=O)C1=NOCC1)C2 c1(C(=O)OCC)cc(Br)c(S(=O)(=O)NC(CN)C(C)(F)F)cc1C Cc1cc(C(=O)NC2CCCC2NC(C2(C(=O)NC3CC3)CC2)=O)cc(C)n1 C1(C(=O)NC(CC)C(C)C)(COC)CCCN(C(=O)CCc2cnco2)C1 N1(C(Cn2c(C)cnc2)=O)CC2(C1)CN(C(=O)CCC(C)(C)C)CC2CO c1(C(N(CCNC(COCCCC)=O)CC)=O)ccc(CC2CC2)nc1C Cc1cnc(C(=O)NC(CN(C(=O)C2=CCSC2)C)Cc2ccccc2)cc1Cl C1(C(C)C)CN(C(C2CC3(CCC3O)C2)=O)CCN1C(c1ccc(F)cc1Cl)=O CC(C)CC(O)C(=O)N1CC(F)(C(=O)Nc2ccc(O)cn2)C1 c1(C(=O)NCCC2CN(C(c3nccn3C)=O)CC(C)O2)cc(F)c(O)c(F)c1 c1(CC(=O)N(CC(C)Cn2ccc(C(F)(F)F)n2)CCO)csc2cccc(F)c12 CC(C)(C(=O)N1CCCC(NC(C2CCC(=O)O2)=O)C1)C1=CCSCC1 N1(C(C(c2ccccc2F)C)=O)CC(C2(NC(C34CC(CO)(C3)OC4C)=O)CC2)C1 N1(C(c2c(C(=O)OCC)c[nH]n2)=O)CC(CNC(=O)C=Cc2ccco2)CC1C C#CCC(C)C(=O)NCCC1CC2C1C(CCCC)SCC(C)C(=O)N2 N1(C(C(C)=C2CCC2)=O)CCC2C(CCCN2C(c2ccc(C)cc2C)=O)C1 Cc1cnc(C(c2nnnn2CCC2(C)CC2)NCCC(C)O)[nH]1 c1(C(=O)OCC(=O)NCCCC)n[nH]cc1[N+](=O)[O-] Cc1nc(S(C)(=O)=O)sc1C(N1CC(CO)C2(C1)CN(C(C1(C)CC1)=O)C2)=O N1(C(C(C)N(CC)CC)=O)CCOCC(C(=O)NC2(CF)CCCC2)C1 N1(C(c2cn3cc(C)nc3s2)=O)CC(CO)C2(C1)CN(C(=O)CC1CCCC1)C2 C(=O)(C#CC(C)(C)CNC(c1c(F)cncc1F)=O)NCC1N(CC)CCCC1 C1(C(N(C2CCCCN(C(=O)CNc3nccs3)C2)C)=O)C2CCC1(C)C2(C)C CC1(C)OCCOC1CC(=O)NC1CCOC(=O)CC1 c1(CNC(=O)NC(C(CC)C)C)c(C)nsc1C c1(C(=O)NC2CC(C)(NC(=O)CCc3nc[nH]n3)C2)ccc2c(c1)COB2O c1(C(N2C(Cc3cn(CC(CC)O)nn3)COCC2)=O)cnc2n1CCS2 N1(CCNC(Cc2cc(C)c(C#N)cc2)=O)CC(C2CCC2)C1c1ccccc1 Cc1[nH]nc2c1CC(C(N1CCC(NC(=O)C=CC(=O)OC(C)(C)C)C1)=O)CC2 N1(C(CC2CC(OC)C2)=O)CCCC2(CNC(=O)CCSC)CCCC12 CC(C)(C)CCCC(=O)N1CCC(C)(NC(=O)C=Cc2ccccc2Cl)C1 n1(C(C)C)cc(CNc2cccc(-c3ccc(CO)s3)n2)c(O)nc1=O N1(C(CN(CC)CC)=O)CCOCC1CCNC(=O)CNC(c1ccccc1)=O Nc1cc(C(=O)NCC2CCCN2C(C2(C(F)(F)F)CC(F)(F)C2)=O)ccc1Cl C1(C(=O)N)C=CC=CC=C1.C1(CNC(CSCC(=O)OC(C)(C)C)=O)CC(C)CO1 C1(C(=O)NC(C(C)(C)C)CNC(c2cccnc2O)=O)CN2CCN1CC2 Cc1cc(Nc2cnc(N3CCOCC3)nc2)ccc1C(C)C(=O)N(C)C c1(NC(C(C)N(C(=O)C(C(C)C)C2CCC2)CC)=O)ccc(O)cc1C C1(NC(CC(C)(C)OC)=O)CCC2(CCN(C(=O)CCc3ccc(C)nc3)C2)C1 C(=O)(CC(C)CN(C)C)NC1CC(CNC(c2cn(CCC)nn2)=O)C1 CCC(C)CCCC(=O)NCCCN(C(c1ccc(F)c(Cl)c1N)=O)C(C)C c1(C(=O)OC)cnc(C(=O)NCC2(CNC(=O)Cc3cc(C)no3)CC2)cn1 Cc1ccc(C(N2CCCN(C(=O)C(C)c3ccon3)CC2)=O)c(Cl)c1Cl C1(CNC(c2cc(C)on2)=O)C2CCC(C2)N1C(=O)C#CC(=O)N1CCOCC1 Nc1c(F)cc(C(=O)NCC2CCC2NC(=O)CSc2ccccc2)cc1F C1(NC(c2scc(C)c2Cl)=O)CC2CC(C1)N(C(c1cc(O)cc(O)c1)=O)C2 C#CCCCCC(=O)NC1CC(F)(CNC(C2CC(O)(C#C)C2)=O)C1 c1(C(N2CCC(CNCCC(F)(F)F)CC2)C)cc(F)ccc1Br N1(C(C(C)=CC)=O)CC2(CCN(C(C3CC3COC)=O)CC2)C1 c1(C(N2C(CN(C(C(n3cc(Cl)cn3)C)=O)C)CCC2)=O)cc(F)c(O)c(Cl)c1 C(=O)(C1=CNC2=NCCCN12)NCCCC(C)NC(=O)CC1=NNC(=O)C1 N1(C(c2cc(CC)sc2)=O)CCCC(N(C(=O)Cc2cn[nH]c2)C)C1 C1(C)(NC(CCc2cc(C)on2)=O)CCN(C(c2csc(C)c2N)=O)C1 C(=O)(C(C)(C)CC(F)(F)F)N1CC(OC)(CNC(=O)C(C)C2CCOC2)C1 c1(CC(=O)NC2(CN(C)C(C3(C(F)(F)F)CC3)=O)CC2)noc2ccc(F)cc12 C1(NC(C2CCCCCS2(=O)=O)=O)CCC12CCN(C(c1cnc[nH]1)=O)CC2 c1(N2CCC(N(CCOC)C(c3snnc3C)=O)CC2)nc(C(F)(F)F)cc(C)n1 N(C(=NCCCc1cccs1)N1CCc2ncsc2C1)CC1(C)CCC(F)(F)C1 c1(C(=O)NCCCCNC(CC(C)OC)=O)cc(Br)ccc1F N1(C(C2C(OC)CCC2)=O)CC(C(=O)N(C2CCSCC2)C)CC(C)(C)C1 c1(CN(C(Cn2cc(C(CC)CC)nn2)=O)C2CCC2)ccccc1Br C(=O)(C(C)(O)C(C)C)NC1C(CNC(CNC(C(CC)CC)=O)=O)C1 Cc1occc1C(=O)NCC1OCCC1C(=O)NC(c1nc[nH]n1)C1CC1 N1(C(COCc2cc(C)no2)=O)CCC(NC(=O)CC2(O)CCCC2)C1(C)C CC(C)C(C)(C)C(=O)NCCC1(O)CN(C(c2ccc(CS(N)(=O)=O)cc2)=O)C1 c1(C(=O)NCC2C(C)(C)CN2c2ncc(Cl)cn2)cc[nH]c(=N)c1N c1(C(=O)NC2CN(Cc3cc(OC)ncc3F)CC2O)cc(F)c(Br)c(F)c1 CC1CCCN(C(c2cnn(CCO)c2)=O)C1CCNC(=O)CC1CC1 c1(C(=O)NCCN(C(c2cc(OCC)c(Cl)cc2)=O)C)c(F)ccc2[nH]ccc12 c1(CCC)nc(C2CC2)ncc1C(=O)NC(C)C.N12CCCCC1CNC2=O C1(OC)(CNC(=O)CCC2CCC2)CCN(C(=O)Cn2ccccc2=O)CC1 c1(C(=O)NCC(CNC(c2n(CC)ccc2)=O)O)c(F)ccc2ccoc12 N1(C(CCOc2ccc(C)cc2)=O)CCC2(NC(c3nc(O)c(C)s3)=O)CC2C1 C1(NC(C2(CC)CCCC2)=O)COC2C(NC(=O)C(C)CC(C)(F)F)COC12 CC1CCN(C(=O)CO)CCN1C(c1cc(CCCO)on1)=O C1(=O)CC(CC)N1C.N1(CC)CCC(NC(=O)C=CCOC)C1 C=CCC(C(=O)NCCCC(C)(F)F)NC(=O)CC(C)SC C(CCN=c1[nH]cc([N+](=O)[O-])cc1C)NCC1CCCN(C(C(CCC)(C)O)=O)C1 Cc1n[nH]c(=NC2CC(F)(CNC(=O)C=Cc3ccc(Cl)s3)C2)o1 CCC(O)C(F)(F)C(=O)N1CC2(NC(c3cccc(-n4cccn4)c3)=O)CC1C2 C(=O)(CCCCSC)N(C(C)CNC(=O)CCCc1ccc(C)s1)CC n1(CCN(C(C2C3CN(Cc4cc(C)sc4C)CC32)=O)C)cnc2ccccc12 c1(OC)ccc(C(N2CC3CN(Cc4ccc(F)cc4I)C3C2)=O)c(OC)n1 c1(OC)cc(C(N2CCCC(CN(C(=O)C=Cc3ncc[nH]3)C)C2)=O)ncn1 Cc1cc(O)cc(=O)n1CC(=O)N(C)CCN(C(=O)C1=CC2CCCC12)C(C)C c1(C(N2CC3N(C(c4c(F)ccc(C)c4)=O)C3C2)=O)cc(O)c(O)c(O)c1 CCC(C#N)C(=O)NCC1CC(COC)CN1C(=O)CCc1cc(C)sc1C c1(O)cnc(CCC(=O)NCC)o1.N1(C=O)CC(NC(=O)OC(C)(C)C)C1 C1(C(N2CC(CC)C2)C)CCC1(C)C C1(NC(C(C(C=C)C)C)=O)C2CC(O)C1N(C(c1csc(C)n1)=O)C2 c1(OC)ccc(C(=O)NCCC(N2CC3CC3(C(N3CCCC3)=O)C2)=O)cc1OC c1(CC(=O)NCCCNC(C(=Cc2ccccn2)C)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NCCCNC(C(CSC)OC)=O)cc(O)nc2cnccc12 CC1CCC(O)C(NC(C2(CNC(c3csc(=N)[nH]3)=O)CCCO2)=O)C1 n1(CC)cc(C(N2CCC(CC#N)C2)C(=O)NCC(=O)OCCSC)c(C)n1 c1(C(C)C)nc(CN(CCCN(C)C(=O)C2CC2)C)cs1 c1(C2(C(N(CC(CN(C)C(c3cccs3)=O)O)C)=O)CC2)ccccc1Cl c1(C(=O)NCC(C2CCOC2)NC(C2(OCC)CC2)=O)cc(S(C)(=O)=O)cs1 Cc1nncc(C(N2CC(C)(NC(C3COCC(C)O3)=O)C2)=O)c1C C=CCCCC(C(=O)NCCOCC1CC1)N1CCCCC1c1cccn1C.OCC N1(C(CCSC)C(=O)NC2CC2)CC(C)OC(C)(C)C1C.C1(C=O)CCC1 C=C(C)C(CC(=O)NCC1C2CN(C(=O)CNS(=O)(=O)CCCC)CC12)OCC N1(C(C(C2CN(C(c3c(CC)ocn3)=O)C2)OC)=O)CCN(C)C2CC12 C1(CNC(C(CC)=CC)=O)COC(C)(C)CN1C(=O)C(=Cc1ccc(F)cc1)C CC(C)(C)C(CNC(c1cccnc1S)=O)NC(=O)Cc1cccnc1Cl C12(CC(N3C4CC(CC(NC(CSC)=O)C4)C3)=O)CCCCC1C2(F)F C(=O)(CC(C)(O)C(F)(F)F)N(CC(C)NC(c1c(COC)noc1)=O)C N1(C(c2cc(C)[nH]c2C)=O)CC2CCC1CN2C(=O)CC1CCCC(O)C1 CC(CC(=O)NC1CN(C(=O)NCCOC(C)(C)C)C1)CC(C)(C)C.C1CO1 c1(C(=O)OC(c2nnc3n2CCCCC3)C)nc2n(c1Br)CC(C(F)(F)F)CC2 N1(C(C(COCC)N)=O)CCC(C(=O)O)(CO)CC1.C1C(=O)N1 CC(C(=O)N1CCOC(CN(C)C(c2ccccc2C2(C)CC2)=O)C1)S(C)(=O)=O C1(CCNC(C=C(C)C(F)F)=O)CCN(C(C2(C)CCCCO2)=O)CCC1(F)F C(=O)(C1=COCCO1)N1CCC(O)(C(C)NC(=O)CCN(C2CCCCC2)C)C1 c1(C(=O)NC2(CN(C)C(c3csc(Br)c3)=O)CC2)cncc2[nH]ccc12 CC(C)(C)C#CC(=O)NCC(C)(c1cccs1)NC(c1cnc(C2CC2)o1)=O N1(CCC)C(=O)CCC1C(=O)NCCC1CCCN(C(=O)Cc2nc(=N)[nH][nH]2)C1 CC(C)C(CN(C)C)C(=O)NC(CNC(=O)C=C1CCC(C)CC1)CC(F)(F)F CC(C)(O)C#CC(=O)NCC1CC(C(=O)NCCc2ccncn2)CO1 C12(CC(=O)NCC3C(NC(CC4CCC(C)(C)CO4)=O)C3)CCC(CC1)C2(C)C Cc1ccc(C(=O)NCC2=CCN(C(=O)CC3CC(C)(C)CO3)CC2)nc1O c1(CCSCC(=O)N(C)CCc2ccccc2)ccc(Br)cc1 c1(-c2cn(CCN(C)Cc3ncoc3C(F)F)nn2)cccc2n[nH]cc12 C1(C2CC2)(C(N2C(C(C)O)CC2)=O)CN(C(=O)CC2CCC(=O)CC2)C1 C(C(C(C)(C)C)NC(=O)C(c1ccccc1F)C1CC1)NC(C1CC(OC)C1)=O C1S(=O)(=O)c2ccc(cc2)C(C)Nc2occc21.Cc1csc(-c2ccsc2)n1 Cc1cnc2c(C(=O)NCC(C)N(C)C(C34COC(CCO3)C4)=O)cnn2c1 CCC(C)C(C(=O)N1CC(N(C(=O)CCc2c(C)noc2C)C)C1)NC(C)=O N1(C(CCOCC)=O)CCN(C(=O)CN(C(=O)C(C)(C)c2ccc(Cl)s2)C)CC1 CCCS(=O)(=O)C(C)C(=O)NCC1CC2CCC(C1)N2C(=O)CC1=NNC(=O)C1 c1(C(=O)NCC2N(C(Cc3scc(CC)n3)=O)CCC2)ccc(F)cc1[N+](=O)[O-] c1(OC)cccc(F)c1C(=O)NCCN(C(=O)CC1CCCS(=O)(=O)C1)C1CC1 CC(C(=O)N(CCCOCCNC(=O)C(C1CCCO1)C1CC1)C)OC C(C)(CNC(c1ccoc1Cl)=O)(CNC(c1ccnn1CCF)=O)OC C1(C(=O)NCCCCN(C(COC(CC)C)=O)CCO)CC(COC)C(OC)C1 CC1(C)C2CCC1(C)C2C(=O)NC1CN(C(c2ccc(CO)s2)=O)CC1C1CC1 S(=O)(=O)(c1cnc(NCCCSC)cc1C)N1CCCC(O)(CC)C1 N1(C(c2c(COC)cccc2)=O)CCN(C(=O)CCCCNC(N)=O)CC1CO C(=O)(C(C)(C)C1CCOC1)NCCN(C(=O)CSCCN(C)C)CCC.CC Cc1noc(CN(C(c2ncc(C(C)C)[nH]2)C(=O)NCC2CCOCC2)C)n1 CN1CCC(C)(CNC(=O)CSCCNC(=O)C(C)(C)F)C1 C1(C(=O)NC2CC(N(C(=O)CC(F)(F)F)C)C2)Cc2cc(Br)ccc2O1 C(CN=c1[nH]c2c(C(=O)OC)cccc2o1)C1N(C(CCCCCOC)=O)CCCC1 N1(C(C(C)C2CCC2)=O)CC2(C)CN(C(=O)CCC3CC3(Cl)Cl)CC2(C)C1 C1(C(=O)NC(C(C(=O)N(C2CCCC2)CCOC)C)C)CC12CCCCC2 c1(OC)cc(C(=O)NCC2C3CC2N(C(=O)CN2CCC(C)C2)C3)ccn1 C1(C(=O)Nc2c(C)ccc(Cl)c2)=CC2=CC=C(C3=CCCC23)C=N1 c1(N(C(CC2CC2)C(=O)NCCCOCCOC2CC2)C)ccccc1 c1(C(=O)NCC2(OC)CN(C(CCC#C)=O)C2)c(OC)ccc2c1CCC2 c1(C(=O)NCC(CO)NC(C2(CC)CC2)=O)c(-c2ccccc2C)noc1C N1(C(c2ccc(SC)o2)C(=O)NC)CCCC1(C)CCc1ccccc1 C(=O)(C1=NN(CCO)C(=O)CC1)NC(C1CN(C(C2(C)CCCCCO2)=O)C1)C CS(=O)(=O)c1ccc(C(N2CCC(F)(CNC(=O)OC(C)(C)C)CC2)=O)[nH]1 Cc1cc(CN2CC(O)CC2C(N2CC3CCC(C2)O3)=O)cc(O)c1 N1(C(c2c(C)cc(C)s2)=O)CC2(CCN(C(C3CCCN3C(=O)C3CC3)=O)CC2)C1 C1(NC(=O)C=CC=C(Cl)Cl)CCCCC1OC(F)(F)F Cc1ncsc1C=CC(=O)NCC1CC1NC(=O)CCCc1ccccn1 C1(C(N2CCC(C)C2c2cn(-c3ccnc(F)c3)nn2)=O)CC2CCC(C1)C2 CCCCCC(C)CC(=O)N1CCN(CCNC(C2(C#N)CCCC2)=O)CC1 C(CCCC(C)NC(c1coc(C2CCC2)n1)=O)NC(c1n(CCC)ncc1)=O CCC(C(=O)N(CC(C)CNC(=O)C(C)(C)c1csc(C)c1)C)NC(C)=O c1(C(=O)NC2CC2)cccc2cncn12.c1(C(=O)NCC(C)C2CC2)cnc(CO)s1 C1(NC(N2C(C(CC)O)CCC2)=O)CN(C(=O)OC(C)(C)C)CC1(F)F C1(F)(C(N(CCC)C2CC2)=O)CCN(C(=O)C=NOC)CC1 C12(CCNC(c3n(CC)ccc3)=O)CCC1CN(C(c1nccc(Cl)c1F)=O)C2 C(=O)(C=C1SCC(=O)N1C)NC1CN(C(CC(C)C(F)F)=O)CC1(C)C C(CCC1CC1)(C(=O)N1CCC(c2nc[nH]n2)C1)NC(c1ccnnc1)=O C(=O)(C(O)C(C)(C)C)NC1(CC(=O)NC(C2CSC2)C)CCCCC1 N1(C(c2cccc(CNC(c3cnn(C)c3Cl)=O)n2)=O)CC2(C)CCC2(C)C1 C1(C2CC2)(CNC(C(CC)n2cccn2)=O)CCN(C(c2cnn(CC)c2)=O)C1 c1(OC)cc(C(=O)NCCC(C)(C)CNC(=O)C2=CCCCO2)c(Cl)cn1 c1(C(N2CCC(NC(C(C)OCC#C)=O)(COC)C2)=O)c(OC)ccnc1O C#Cc1cccc(C(=O)NCC(F)CNC(=O)C(C)n2ccnc2)c1C c1(C(N2C(CC)CN(C(=O)CCC3CCCCO3)CC2)=O)cc(O)cc(N)c1C C(CCOC1C(OC)C1C)(C(=O)N1CCCC1C)NC(C=CC)=O.C1(=CC)CC1 CCC(C)(C#N)C(=O)NC1(C)CCCN(C(=O)C(C)(C)Oc2ccc(Cl)cc2)C1 C(=O)(C1=CCC2CCC1N2C(=O)OC(C)(C)C)NC1CC(C)Sc2c1ccs2 N1(C(C2C(C)CCC2)=O)CC2=C(C1)CN(C(c1ccc(O)c(Br)c1)=O)C2 CC12OCC(CSCC3CCCCO3)(CO1)CO2 CC1=C(C(=O)N2CCCC2CN(C(=O)CNC(c2ccc(C)s2)=O)C)CCCO1 N1(C(c2ccnc(C)n2)=O)CCOCC(NC(=O)C(C)OC2COC2)C1 C1(NC(c2c(C)cncc2C)=O)CCC(O)CN(C(=O)C(n2cc(Cl)cn2)C)C1 Cc1cc(C(=O)NC2CN(C(=O)CCC3CCCCCC3)CC2C)c(C)o1 N1(C(CCCNC(C2(COC)CCCC2)=O)=O)CCCC(O)(CO)C1 CC(S(=O)(=O)Cc1ccc(C2CCCCC2)o1)C1CCOCC1 CN=C(NCCCOCC(=O)OC)NCCC1CCC(C)O1 N1(C(CCSCCC)=O)CCN(C(C2CN(C)C2)=O)C(CC)C1 N1(C(CC(C)C(C)(C)NC(=O)C(CO)C(F)(F)F)=O)CCC2(CC1)CC(O)C2 CCCCC(CNC(C1(C(=O)OC)CCCO1)=O)NC(C12CCN(CC1)C2)=O N12CCCC(c3nnnn3C3(C)CC3)(C1)NC(CSC)C2=O.N(C)(C)C(C)=O c1(OC)c(C)cc(C(=O)NCCN(C(=O)Cc2ccc(C)c(F)c2)C)cc1Cl C(=O)(C(N)CCC(N)=O)NCC12C(N3C(C)(C)CC3)CC(C1)C2 CCCCS(=O)(=O)NCC(=O)NC(CNC(C1CCC(=O)C1)=O)CC(C)C c1(-c2cn(CC(=O)NCC3C(C)C3C)nn2)ccc(C(=O)O)c(F)c1Cl c1(OC(C)C)cccc(C=CC(=O)NC(C)CCN(C(=O)COC(F)F)C)c1 c1(CNC2CCC(C(N3CCCC(C)C3)=O)CC2)csc2ccccc12 N12CCN(C3CCCC13)C(=O)C1CC(C1)OCC2=O.c1(OC)cc(OC)[nH]n1 C(C(C)(C)C(C)(C)O)NC(C(CC)N(C)C(c1ccccc1)=O)=O c1(CNC(C2CN(c3c(OC)cncn3)CC2C#N)=O)cc(F)cc(Br)c1F Cc1ccc([N+](=O)[O-])c(N2CCC(C)C(NC(C3(C)CCC3)=O)C2)c1 c1(SCC(=O)NCC2C(CNC(C3CCC(C)O3)=O)C2)ccc2ccccc2c1 C(=O)(CCC(F)(F)CCO)N(Cc1ccc(OC)cc1)Cc1ccccc1 N1(C(c2nc(OC)c(F)cn2)=O)CCC2(CCC2NC(=O)Cc2ccon2)CC1 Cc1cc(C2CC2)ccc1C(=O)NCCNC(=O)CCCN(C)C1CC1 N1(C(c2cccc(C)c2N)=O)Cc2[nH]nc(C(=O)NC3CCN(C(C)C)C3)c2C1 C1(CN(C(C(CC2CC2)OC)=O)C)CCCN(C(=O)C(c2cnn(C)c2)=O)C1 C(=O)(CC(C)CC(C)C)NC1C2CN(C(C=CCOC)=O)CC1C2 C=CC(C)(C)C(=O)OCC1CCCC1C N1(C(c2oc(C)c(CO)c2)=O)CCOCC(CNC(=O)CC(C)(C)O)C1 C(=O)(C1=CCOCC1)N(C1CCN(C(CCC(=C)C)=O)CC1)C.N12CCCC1C2 C(C)(CCNC(C1(C)CC1C(F)(F)F)=O)NC(C=CCOC)=O N1(C(CCOCC#C)=O)CCC(C)(CNC(=O)CC2(O)CCCN(CC)C2)CC1 n1(CC(N2C3C(NC(c4cc(Cl)cs4)=O)C(C3)C2)=O)ccc2cc(F)ccc12 C(N=c1[nH]c2c(c(=NCC3CCC4CC34)[nH]1)CCCC2)c1ccc([N+](=O)[O-])c(Cl)c1 N1(C(=O)C=CC2CCOCC2)CC2CCC(NC(=O)COc3ccsn3)(C2)C1 c1(C(=O)NC2CC(NC(CCC3CCC(C)O3)=O)C2)csc(N=S(C)(C)=O)n1 C#CCCN1C(=S)NOCC2CC3CC(C3C2)OC1=O.c1(CO)ccccc1 c1(C(=O)NC2C(CNC(=O)CN3CC4CC4C3)C2)cc2ccncc2[nH]1 C1(NC(C(CSC)C)=O)CCN(C(c2sncc2C)=O)C12CCC2 C12(NC(Cc3cccc(CC)c3)=O)CCN(C(=O)CC3(C)CCC3)CC1C2 CN1CCCC(C(=O)NC2C=CCCC2CNC(c2cncn2C)=O)C1 Cc1cc(C(N2CCC(NC(C3(C)C=CCCC3)=O)C2)=O)ncc1CO c1(-c2nc(CCC(C)C)nn2Cc2ccsc2)ccc2nnnn2c1 N1(C(c2ccc(OC)cc2O)=O)CC2CC1CN(C(C1CC1C(C)C)=O)C2 c1(C(=O)NCC(CC(C)C)NC(=O)CCN2CCC2)cc(S(N)(=O)=O)ccc1O CC1CCCC(CO)(N)CC1.C1(=C2CCSCC2)CCSCC1 C1(NC(C(c2ccc(C3CC3)cc2)N)=O)CCOC(c2cccnc2)C1 c1(CC(=O)NC2CN(C(C(CC)CC)=O)C(C)C2)[nH]c(C(=O)OC)c(C)c1C(C)=O CC1(C)CCN(C(C2CC2(Cl)Cl)=O)CC1NC(c1coc(C2CCCCC2)n1)=O C(N=c1[nH]c(Cl)c(C#N)s1)C1CCC(CNC(C2(C)CCCNS2(=O)=O)=O)CC1 C12(NC(c3cc(Cl)no3)=O)CCC(C(F)(F)F)(CC1)C2.C12CC3CN(CC13)C2=O c1(NC(C(=O)Nc2cn(CC)nc2)=O)cc(Br)cnc1OCC(C)C C=C(Cl)CCC(=O)NCC1(C)CCC(NC(c2nc(O)c(C)s2)=O)C1 Cc1cc(Br)ccc1-n1cc(C(N2CCN(C(c3ccccc3)C)CC2)=O)nn1 c1(OC)ccc(C(N)=O)cc1C(=O)NC1CC(CNC(c2cc(Cl)n(C)n2)=O)C1 Cc1ccn(C)c(=O)c1NC(=O)C(Cn1cncn1)NC(C1CCCN1C)=O C(=O)(C(Cc1ccccc1)C(F)(F)F)N1CC(C)(NC(C2(F)CCOC2)=O)C1 C12(NC(C(C)=C3CC3)=O)CC3CC(C1)CC(NC(C1CCCC(O)C1)=O)(C3)C2 C(=O)(C1Cc2ccccc21)N(CCN(C(C1CC(C)(CC)C1)=O)CC)CC CC1(C)CC(CC(N2CCCC2C(=O)NCCCCC2CC2)=O)CCO1 CN1CCC(C(N2CCN(CCN(C(=O)C(F)C(C)(C)O)C)CC2)=O)S1(=O)=O c1(C(N2C(NC(C3CN(C(C(=O)OCC)C)C3)C)CCC2)=O)cccc(C)c1F C12(CCNC(C3CNC(=O)N3)=O)CCC(CC1)N(C(=O)C(O)C(F)(F)F)C2 N1(C(C2(CCC=C)CN(C(=O)C#CC(C)C)C2)=O)CC(C)OC(C)C1 CC1(C)CC(NC(=O)C=CCNC(C23CCCC2C3)=O)C1 c1(CC)cc(C(=O)N(C)CCN(C(c2cnc(C3CCOC3)s2)=O)C(C)C)ncn1 C1(NC(C2C(OCC)CC2)=O)CN(C(=O)Cc2cccc(O)c2)CC12CCCC2 N1(CCCC)CCOCC1C(=O)NCCCCNC(=O)C(C1CC1)C1CC1 Cc1c(CC(=O)NC2CCC(C(=O)N(C3CSC3)CCO)C2)ncn1C CC(CC(C)(C)C)C(F)C(=O)NCCCCCN(C)C(c1cc(C2CC2)on1)=O c1(OC)ccccc1NC(=O)CCNCc1cc(CC#N)on1.C(C)=O C1(NC(COC)=O)CN(C(c2cc(C(F)F)nn2C)=O)CC1SC C(=O)(CCC(CF)CF)N1C2CC(C(=O)NC(C(N)=O)C3CCCC3)(OC2)C1 c1(N(C)CC)ccc(C(=O)N(C2CN(C(=O)CC(C)C3CCCO3)C2)C)cc1 N1(C(c2cc(C3CC3)nn2C)C(=O)NCC(=C)C)CCCCC1C c1(OC)cc(NC(c2nc(CC3CC3)no2)C)[nH]c(=N)n1 N1(C(c2c(C)ccnc2C)=O)C2CCC1CN(C(c1nnc(Cl)cc1N)=O)C2 CCCCCCC(C)C(=O)N1CCOC(C(=O)NCCc2c(C)n[nH]c2C)C1 CCCC(C)(CO)NC(=O)CCCNC(=O)CC1OCCC1(C)C C12(C(N3CCC(CNC(CC(C)C(F)F)=O)C3)=O)CCCC(CCC1)C2 CCCC(C(O)C(=O)N(C1COCC1OC)C)NC(c1cccc(CC)n1)=O c1(C(=O)OCC)cccc(Cl)c1N(C(c1ccc(F)cc1)=O)CC1CCC(=O)N1 C(C(C)NC(=O)CCc1c(C)noc1C)(C(C)C)NC(Cc1cn(CC)nc1)=O N1(C(c2cnc(CC)s2)=O)CC(N(C(=O)C(C(C)C)C2CCC2)C)C2(CC2)C1 Cc1ccc(O)cc1C(N1CC(N2CC3COCC3C2)C1)=O.C12CCC(CC1)S2 CC1CN(C(=O)CN2CCC2)CC1NC(c1ccc(-c2cc[nH]n2)s1)=O c1(OCC)ccc(CC(=O)NCC(O)CNC(C2(C)CC2(C)C)=O)cc1 c1(C(=O)NCC(CC)NC(C2CCC(=O)O2)=O)oc2ccc(OC)cc2c1C C1(C(=O)NCCOCCCNC(c2cc(C)c(Cl)s2)=O)CC2(C1)CC(F)C2 CCCCCC(C)CC(=O)NC1CCN(C(c2ccn3cccc3c2)=O)C1(C)C C1(C(N2C(C)CCC2)=O)CCC(C)N1C(=O)C(Cl)Cl c1(C(C(OC)OC)NC(=O)Cc2ccccc2)ccc(C)cc1 C1(C(N(C)CCOCCNC(=O)Cc2ccns2)=O)CC2(C1)CC21CCC1 c1(CNC(C2N(C(C(C)CC3CC3)=O)CCC2O)=O)cnc2n1CCC2 C1(NC(CCCC(N)=O)=O)CCCCC12CCN(c1ccc([N+](=O)[O-])c(O)n1)C2 N1(C(C(C)C2(O)CCC2)=O)CCC2(CC2)CC1C(=O)NCC(F)F c1(C(N2CCC(O)(CNC(c3c(C)cc(C)s3)=O)C2)=O)ccc2nn[nH]c2c1 c1(C(=O)NC2C(NC(c3cn(C4CCC4)nn3)=O)C2)[nH]cc2c1CCCC2 C1(C)(CC(=O)NCC(COC(C)C)O)CCN(C(=O)CC2CCCC(=O)C2)C1 C(C(C)(O)C(=O)N1CC(CNC(c2cccc(OCC3CC3)n2)=O)C(C)C1)OC N1(C(CC(C)SC)=O)CCN(CCN(C)C(c2c(C)ncn2O)=O)CC1 N1(C(C(CC)COC)=O)CCC(O)C(C(=O)NC2CCCCC2CO)C1 c1(C(=O)OC)cccc(C(N2CCC(O)(CNC(C34CC(O)C3C4)=O)C2)=O)n1 N1(C(=O)NC(c2nc(C3CC3)n(C)n2)C)CCC2OCCC2C1 c1(C(=O)NCC(C2CCCN2C(C2CCCC2)=O)C2CC2)cc2ccncc2s1 c1(CNC(CCSCC)=O)ccc2c(c1)CCCC2NC(=O)C=C1CCCCC1 C(=O)(C(CNC(=O)C(=O)NCCOC)C(C)(C)C)NC1N(CCC)CCC1 Cc1nc(C2CN(C(=O)C(Cn3cccn3)NC(=O)CC(C)C3CC3)C2)n[nH]1 c1(C(=O)NCc2ncc(-c3ccn(C)n3)cn2)ccc(Cl)c(Br)c1 c1(C(=O)NC2(CCNC(=O)C=CC3CCOC3)CC2)cc(O)cc(F)c1 c1(CC(=O)NCC2CC2)ccc(CC2N(C(=O)CNC(=O)C3CC3)CCC2)cc1 c1(C(=O)NC2CC2CNC(c2ccoc2C(F)(F)F)=O)cc(O)nc(Br)c1 CCCC(C)(C)C(=O)NCCOCCN(C)C(C1(CO)CCC1)=O N1(CC(=O)NCC2CCN(C(c3cnsc3)=O)C2)CCS(=O)(=O)CC1 C1(NC(Cc2cnn(C)c2C(F)F)=O)COCCN(C(C2CC(=O)CO2)=O)C1 n1(CC)nc(C)c([N+](=O)[O-])c1NCC1CN(C(=O)C2=CCCCC2)CCC1C N1(C(Cn2nnc(C)n2)=O)CCOC2(C1)CN(C(=O)C(C)C(F)F)C2 N1(C(CC(COC)NC(c2sccc2CO)=O)=O)CCC(N=[N+]=[N-])C1 c1(CCC(=O)NC2CC(NC(=O)CC34COCC(C3)C4)C2)ccccc1Cl C1(NC(=O)OC(C)(C)C)CN(C(=O)Nc2cccc(-c3ccc[nH]3)c2)CC12CC2 c1(C(N(CCCCCC)CCNC(=O)CCC2(C)CC2)=O)cnn(CC)c1C C#CC1(C(=O)NC(C)CCNC(=O)CCNC(c2ccccc2)=O)CCC1 c1(OC)ccc(OC)c(C=CC(=O)NCC2(F)CCC(NC(C3CC3F)=O)C2)c1 c1(C(=O)NCC2CC(NC(CN(C(C(C)C)=O)C)=O)C2(C)C)ccc2sccc2c1 N1(C(c2c(CC)onc2)=O)CCN(C(c2cncc(F)c2)=O)C(C(F)F)C1 O=C(CC1CCc2ccccc21)NC1CC(F)CN(C(C2(CC3CC3)CCC2)=O)C1 CC1CCCC(C#N)(N(C(C2(C3CCCO3)CCC2)=O)C2CC2)C1 Cc1ccc(OCCC(N2CCC(C(C)NC(=O)Cn3cncc3C)C2)=O)cc1 C1(CCC)CN(C(=O)C(CCO)N(C)C)CCN1C(=O)CC1(O)CCCCC1 C(=O)(C1=Cc2cc(F)ccc2OC1)NCC(C)NC(C1CC(C)(F)C1)=O c1(C(C)C#N)ccc(C(=O)NCCN(C)C)cc1.C12(F)CN(C1)C2=O c1(CN2CCCC(C(=O)Nc3cccc(F)c3O)C2)c(Cl)[nH]c2ccccc12 c1(C(C)C)ccc(C(N2CC(C3CCN(C(C=CC(=O)NC(C)C)=O)C3)C2)=O)o1 c1(CNC(c2cccc(C(=O)NCCN=[N+]=[N-])c2)=O)cc(C(=O)OC)ccn1 C1(C)(C(N2CC(=C(CNC(C(C)Cn3ccnc3)=O)F)C2)=O)COC(=O)C1 CC1(C#CC(=O)N2CCC(C)(C)CC2C(=O)NCC2CC(F)(F)CO2)CCCO1 C1(NC(C(OC)OC)=O)CCSC12CN(C(C1CCCC3(CC3)C1)=O)C2 C(=O)(C(F)CCC(C)C)N1CC(C(C(=O)NCC2(C)CCC(=O)N2)OC)C1 C=C(C)CC(C(=O)NCc1cccc(CN(C(=O)COC2CC2(F)F)C)c1)OC CC1CN(C(c2csc(Cl)c2Cl)=O)CCCN1C(=O)CC1=CCCCC1 C1(C(=O)NC(CC(C)C)(C)CNC(=O)C=CC2CCC2)CCC2(CCC2)CC1 N1(C(c2c(C)nc(COC)s2)=O)CCCC1C1CCCN1C(=O)CSCCOC c1(Nc2c(OC)c3c(cc2)CCC3)ccc2c(c1)CC(C(=O)O)CCC2 CCCCCCC(C)C(=O)NC1CCC(NC(c2cc(C#N)c(C)cn2)=O)CC1 Cc1ccc(C(=O)NC2CC3CC2N(C(c2cccc[n+]2[O-])=O)C3)cc1CO c1(C(c2ccc(OC)cc2)O)n[nH]c(=NC(=O)NCCC#N)s1.C1(=O)CCN1 N(C(=NCCCOC(F)F)NCC(C(F)F)C1CC1)CC(C)(C)F Cc1ccc(N)c(C(=O)NC(CO)C(C)NC(c2cn(C3CC3)cn2)=O)c1F N1(C(C(C)=CC2CC2)=O)CCCCC(NC(c2cnc(C(F)F)cn2)=O)C1 CC1CC(NCc2cc(F)ccc2C(F)F)CCN1C c1(CNc2c(C(=O)Nc3c(I)ccc(C)c3)ccc(Cl)n2)cc(F)c(C)c(F)c1 Cc1[nH]nc(C(F)(F)F)c1C(=O)NC(C)CNC(C1(C)CCC(=O)N1)=O c1(CC(=O)NCC(CC=C)NC(C23CCC2C3)=O)noc2ccccc12 CC(C)(F)C(C)(F)C(=O)N1CC2CC1(c1cn(CCC3CC3(Cl)Cl)nn1)C2 C(C(C(=O)NCC(C)(O)C(F)F)C(C)C)NC(c1n[nH]c(C)c1Cl)=O N1(C(C2(CC=C)CN(C(c3cscc3OC)=O)C2)=O)CC(C)=CC(C)C1 N1(C(CC=CCC)=O)CCC(C2(O)CN(C(=O)Cc3ccc(C#N)nc3)C2)CC1 CC1CCN(C(c2cccc(F)n2)=O)CC1NC(C12CCC(CO)(CC1)C2)=O c1(C(C)NC(c2cnc(Cl)s2)C)cncc(Cl)c1 c1(C(N(C(C)CNC(=O)C=C2CCCCC2)C)=O)cc(Cl)ccc1O c1(CC(=O)N(CC(C)NC(=O)CC2CC(N(C)C)C2)C)ccc2c[nH]nc2c1 C1(CNC(C2(CC#C)CC2)=O)(COC)CCN(C(=O)C(C)CO)C1 N1(C(C(CC)OCC)=O)CCN(C(c2ccc(C)c(O)c2)=O)C(CC(F)(F)F)C1 c1(C(N2CCC(n3c(C)cnc3)CC2)=O)cc(Br)ccc1OCCN n1(CC(=O)NC(C)COC(C)(C)C)cc(CCC2CCCCC2)nn1 N1(C(CCNC(N)=O)=O)CCC(CO)(SCC(=O)NCC2CCCO2)CC1 c12cccc(c1)N1CCN(CC1)C2.c1(-n2ccc(C(C)(C)C)n2)ccccc1F C1(C(N(CCCN=[N+]=[N-])C)=O)CC2CC1CN(C(C1C3C4CCC(C4)C13)=O)C2 O=C(CC1=CCN(C(c2cncs2)=O)CC1)Nc1cccc(Cl)c1O c1(CN2CC(C(=O)Nc3ccns3)C(O)CC2)cccn2ccnc12 CC1CN(C(c2cc(C3CC3)no2)=O)CCC12CCN(C(=O)C(C)C1CC1)CC2 c1(C(=O)NC(C)CC2COc3ccccc3O2)ncc(Br)c(=NC2CCCCC2)[nH]1 N1(C(=O)OC(C)(C)C)CC(OC(N2CCCCC(C)(F)C2)=O)CCC12CC2 N1(C(C)C)CCN(CCC(N2CCN(C)CC2)=O)CC1CC(F)(F)F c1(C(C(=O)NCC(C)C)N(CCC)CCNC)cccc(C(=O)N(C)C)c1.OC c1(CC(CNC2CCCC3CC23)NC(N2CCCC2)=O)ccccc1Br C1(C(=O)OC)CCN(C(=O)C2N(C(=O)CC(C)SC)CCC2(C)C)O1 N1(C(COc2cc(C)on2)=O)CCC(CC(=O)NCc2cocn2)CC1 C1(C(=O)NC(C(C)N(CC)CC)=O)CC1(C)C(=O)NC(C)C CC1Cc2nc(Cl)nc(N3CCCC(n4ccnn4)CC3)c2C1 CCC(O)C(C)C(=O)N(C1CC(O)C1)Cc1ccccc1.C12CN(C1)C2=O C(=O)(CC(=O)N1CCCC1CN(C)C(c1cc(CC)[nH]n1)=O)OCC N1(C(c2cc(C)n(C)n2)=O)CCOC2CCN(C(c3cc(F)n(C)n3)=O)CC12 Cc1sncc1C(=O)NC1(CNC(c2cnc(O)s2)=O)CCOC1 N12CCCCC1C2C(=O)NC1CC(C(=O)OC)C1.c1(OC)ccccc1 N1(C(c2c(C)snc2)=O)CCn2ncc(CNC(=O)CNC(C3CC3C)=O)c2C1 c1(N2CCCC(C)(C)CC2)nccc(=NCCCNC(=O)C2CC2)[nH]1.C(N)(=O)N C(=O)(CCCC(C)=O)NCc1cc(C(=O)NCCCCC)no1 C(C(C)(C)C#CC(=O)NCCN1CC2CC2C1)NC(CCC1CC(C)C1)=O C1(NC(c2ccc3c(c2)OCC3)=O)CN(C(=O)Cc2cscn2)C2(CCOC2)C1 C(=O)(CCCCCC(C)C)NCC(C(=O)N(CC)CC1CC1)N(C)C C1(NC(C=C(C)C)=O)CN(C(c2ncncc2Cl)=O)Cc2ccnn2C1 c1(OCC(=O)NCCC(C)NC(=O)C(C#N)C2CC2)cnc(Cl)cn1 Cc1cc(C(C)C)c2c(C(C)NCCCn3cnc4ccccc34)noc2n1 C1(CC=C)(NC(=O)CC(C)SC)CCN(C(=O)C(C)C#N)C1 C1(OC)CN(C(c2cccc(O)c2)=O)CC1C(=O)NCc1ccncn1 c1(C(C2CC2)NC(=O)NCC2(O)CCCCCC2)cc(Cl)ccc1Cl c1(NCc2cc(OC)ncc2)cc(S(=O)(=O)N2CCCC(CF)C2)ccc1C#N c1(C(N(CCCN(C)C(c2cc[n+]([O-])cc2)=O)C)=O)[nH]nc2c(=O)n(C)cnc12 c1(C(=O)NCCOCCCC)occc1C(=O)NCCNC(=O)C(CF)CC c1(C(N2CC3C(N(C(C(F)=C(C)C)=O)C)C3C2)=O)cc(F)cc(Cl)c1 CCC(C(=O)NCC1CN(C(C2(C(C)(C)C)CCC2)=O)C1)C(C)C c1(CC)onc(C(=O)NCCC(C)NC(C2CCN(C3CCSC3)CC2)=O)c1C CCCCCC(O)C(=O)N1CCCC1C(=O)N(CC)CC1CC2CCC1CC2 N1(C(Cn2ncn(C)c2=O)=O)C2CCC1CN(C(c1ncc(Cl)s1)=O)CC2 C(=O)(C(CC(=O)NC(CNC(c1cc(Cl)cc(Cl)c1)=O)C(C)C)C(C)=O)OCC Cc1c(C(=O)NCC2CC(NC(C3CCCOCC3)=O)C2)cnn1C n1(C(C(=O)NC2C(CC)CN(C(C3(CF)CC3)=O)CC2)C)cc([N+](=O)[O-])nc1C c1(C(N2CCC(CC#C)(C(=O)O)C2)=O)ccc(Br)c(F)c1.C(C)(C)C c1(C(N2CC(CNC(c3c(COC)scc3)=O)OCC2)=O)cccc2oncc12 Cc1oc2ccccc2c1C(=O)NC1CN(C(C2CC(S(C)(=O)=O)C2)=O)C1 C1(C(=O)NCCCN(C)C(c2cnnn2C)=O)CCC12CCCO2 N1(C(c2c(C)ncs2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1c1ccccc1Cl C1(C(N2CCC(C(C(=O)N(CC(CC)C)C)(C)C)C2)=O)CC2(CC(=O)C2)C1 C1(CC)CCCCC1NC1(C)CN(C(=O)COC2(C)CCOCC2)C1 C(=O)(C(C)(F)C(F)(F)F)NCCOC1CCN(C(CC=C(C)C)=O)CC1 CC1=CCC(C)(C(=O)NCC2(C)CCN(C(=O)CSCc3ccccc3)C2)CC1 C(C)(CCC(=O)NCCC1CCCOC1)NC(c1cn(CC=C)nc1)=O c1(C(N2CC(O)CC(NC(n3c(C)csc3=O)=O)C2)=O)cccc2c1C(=O)NC2 C(C=C(Cl)Cl)NC(C1C(C(C)O)C1)=O C(=O)(CCC(C)(F)F)NCC1(F)CCN(C(C(CCC)C)=O)C1 c1(C(N2CCC(O)(CCNC(C3(CC4CCC4)CC3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] N1(C(CCn2c(C)nc([N+](=O)[O-])c2)=O)CCN(C)c2ccc(Cl)cc21 C(=O)(C(C)=Cn1ccnn1)N1CC(N(C(C2(COCC)CCOCC2)=O)C)C1 N1(C(Cn2c(C)nnn2)=O)CC(NC(c2n[nH]c3c2COC3)=O)CC(C)(C)C1 Cc1cc(C(=O)NCC2CC(NC(CNc3ccc(CF)cc3)=O)C2)cc(Cl)c1 CCC(O)C(C)C(=O)NCC1CC(O)(CNC(c2cccc(CC#N)c2)=O)C1 C1(C)(C(N(CC(n2cccn2)C)CC(C)C)=O)CCCN(C(C)C(C)(C)C)C1 C1(C(N(CC=CC(=O)N(CC(CC)O)C)C)=O)CC2CC1CC2=O C1(CNC(CCN(C(=O)CC(C)n2ccnc2)C(C)C)=O)OC(=O)NC1(C)C N1(C(c2nn[nH]c2Cl)=O)CCN(C(c2cc3cccnn3c2)=O)C2(CC2)C1 C(CNC(c1ccc(=N)[nH]c1)=O)(C(=O)NOC1CCC1)N(C)C C12(CNC(c3ccc(C)s3)=O)CCC(C1)N(C(c1ccc(Br)o1)=O)C2 c1(NC(c2ccc(F)c(Br)c2)=O)cccc(F)c1C(=O)Nc1cnc(Cl)cc1I c1(C(N2CCCC(CN(C(C3(C)ON=C(C)C3)=O)C)C2)=O)c(C)nn(C)c1Cl C(=O)(C(C)C1=CCCC1)NC(CNC(c1c(F)ncc(OC)c1)=O)C C12(CCNC(N(CC(C)(C)OC)C)=O)CCC1CCN2 c1(CNC(=O)NCC2(c3cccnc3Cl)CC2)c(C(F)(F)F)cccc1Cl N1(C(c2c(C)coc2)=O)CC(NC(c2cnn3c2OCCC3)=O)CCC(O)C1 N1(C(C=C(CC)CC)=O)CC2(CCCC2)C1C(N1CCCC(CN=[N+]=[N-])C1)=O C(=O)(CC(C)C(F)F)NCC1C(C(N2C(COC(C)=O)CCC2)=O)C1(C)C N1(C(c2ccc(CN(CCC)C)o2)=O)CCC(CO)C(C(=O)O)C1.c1(N)nccs1 N1(C(CCSC)=O)CCCCC1C1CCN(C(c2ccc(O)nc2)=O)C1 CON(C)CCN=c1nc2sccc2c(N2CC3CCCCC3(N(C)C)C2)[nH]1 N1(C(C(C(CC)C)O)=O)CCC2(CCOCC2)C(NC(c2ncn(CC)n2)=O)C1 N1(C(CSC)=O)CCC2(CC1)CC2CNC(c1cc(C(F)(F)F)n(C)n1)=O N1(C(CC(C)(C)O)=O)CCN(C(c2cn(C3CCOC3)nn2)=O)CC1C1CC1 C1(NC(c2c(C)nc(COC)s2)=O)CN(C(c2occc2C)=O)CC2(CCC2)C1 C1(C(N(CCSC)C)=O)CN(C(=O)C(C)(C)C)CC1(F)F N1(C(CN(CCOCCOC)C)=O)CCC(C)(C)C1.C(C(=O)NC(C)C)O c1(OC)ccc(CC(=O)NCC2CN(C(C3CCCOC3C)=O)C2)c(C)c1 C12(CCNC(Cc3c(C)nsc3)=O)CCC(C1)N(C(c1cc(C(N)=O)co1)=O)C2 C1(C(=O)NC(C)(C)CC(=O)NCCC2(C)CC2(F)F)COCC1C(N)=O c1(OC)cc(CNCCC(C)S(C)=O)cc(Br)c1 c1(C(N(CC(C)NC(=O)C(=O)c2ccco2)C)=O)cc2c(F)c(F)ccc2[nH]1 CCC(CCCC(=O)N1CC2CCC2(C)C1)NC(c1cnnn1C)=O n1(CCN(C(=O)C(N2CCNCC2)C2CC2)c2ccco2)cc(Cl)cn1 C1(CNC(=O)N(C2CCCC2OC(F)F)CC2CCCO2)CCCCC1 CCCCC(CC)CC(=O)NC1CCCN(C(=O)Cc2cc(Cl)sc2Cl)C1 c1(C(=O)NCc2cccc(NC(COC)=O)c2)ccc2c(c1)OC(C)(C)C2 Cc1nc(C)c(C(=O)NCC2CC2CC(=O)NCC2CC23CC3)s1 N1(C(C2ON=C(C(C)C)C2)=O)CCC2(CC1)CCN(C(C1CC(=O)N1)=O)C2 C1(C(N2CCC(CNC)CC2)=O)Cc2ccccc2C1 Brc1ccsc1CN1CC(c2nncs2)C1 N1(C(C2CC(O)(CNC(=O)CC(F)(F)C(F)F)C2)=O)CCCC2(CCOC2)C1 C1(C)(CC(=O)NCC(C)CC2CCCC2)CCN(C(=O)C=Cc2cc[nH]c2)C1 CCCC(C)(O)CC(=O)NC(C)(C)CC(=O)NC(C)C(=O)N(C)CCOC c1(C(N2CCC(O)(CCNC(C(C)=CC3CC3)=O)C2)=O)ccccc1P(C)(C)=O c1(C(=O)NCC2(F)CC(CNC(C(F)OC)=O)C2)ccn2c(C)cnc2c1 N1(C(Cc2c(C)cc(Cl)nc2)=O)CCCN(C(C2CC(CF)C2)=O)CC1C(C)C c1(C(=O)OCC)cc(N2CCC(CN(C)C(c3cnncc3O)=O)CC2)ncn1 N1(C(C(CN(CC)CC)F)=O)CCC2CC1CN(C(=O)CCN(C)C(C)=O)C2 C1(CS(=O)(=O)NC(c2cc(CNC(C)=O)on2)CC)CCC(=O)N(C2CC2)C1 c1(CC)nc(C(C)NC(c2nnnn2-c2ccccc2)CC)no1 C(=O)(C1=CC2CCCCC12)NCC(CC)NC(c1ccc(F)cc1C(F)F)=O c1(C(=O)NCC2N(C(C=C(CC)CC)=O)C3CCC2C3)ccc2ccccc2n1 c1(C(N(C)CC2CC(F)CN2C(=O)C=CC(F)(F)F)=O)cccc2[nH]ncc12 c1(C(N2C(C(=O)Nc3c(C(N)=O)cccc3)CC3CC32)=O)ccc(O)cc1Cl c1(C(=O)NCC(CC)NC(C(CC#C)O)=O)c(C)ccc(F)c1N CC1=C(C(=O)N2CCCCC2C(C)(C)CNC(=O)C(C)C2CCCO2)CCO1 N1(C(C2CC(CC)C2)=O)CC2(C=C(C(=O)N3CCC(CO)C(C)C3)CO2)C1 c1(C(N2CCC(N(C(=O)COCCOC)CC)C2)=O)cnc2ccccc2n1 CC(Cc1cnn(C)c1)C(=O)NC(C)(CNC(=O)Cn1cnc(Br)c1)CO C1(NC(CC(=O)NCC2CC2)=O)CN(C(=O)CCC2CCCO2)CC1C(F)(F)F n1(CC)ncc(Cl)c1C(N1CC(NC(c2cscc2OC)=O)C(C)C1)=O c1(OC)cc(CN2CC(F)(C(=O)NCc3c(Br)cnn3C)C2)cc(Br)c1O CC1CCCCC1(C)C(N1CCC(C)(C(=O)N(C)Cc2cccnc2O)CC1)=O N1(c2nnc(-c3ccn(C)c(=O)c3)n2CCOCCO)CCc2ccc(F)cc2C1 CON(C)C(=O)C(C)NC(C1(CO)CCCN(C(=O)C(C)NC(N)=O)C1)=O c1(NCCN(CCCC)C)[nH]c(=NCCc2cc(F)cc(F)c2)nc2sccc12 c1(C(=O)OCCCC=C)nc2nccc(C)n2n1 Cc1nc(CC(=O)NCC2(NC(c3oc(C)cc3C)=O)CCC2)c(Cl)s1 NS(=O)(=O)c1ccc(-c2nc(-c3ccc(O)cc3F)no2)cn1 c1(C(c2nnnn2C2CCC2)CC(C)SC)noc(-c2cccn2CCCF)n1 c1(CC(=O)NC(CNC(C(N2C(=O)CCC2=O)CC)=O)CO)ccc(C#N)cc1 N1(C(COCCCCC)=O)CCCCC1C1CCN(C(=O)CC(C)COC)CC1 N1(C(C2(CC#C)CC2)=O)CCCCC(NC(=O)C(Cc2cnc[nH]2)NC(C)=O)C1 C(=O)(N=c1cc(C2CC2)n(C(C)C)[nH]1)C1(C)CCN(C(C(C=C=C)C)=O)CC1 c1(C(=O)NCC(C)CN(C)C(C2(C)CCCC2)=O)cnnc(O)c1 CC(C)C(C(=O)NCC1CCCCC1NC(c1nc(C)n(C)n1)=O)NS(N)(=O)=O C1(N(C(=O)C(F)(F)C2(O)CCC2)C)CCC(NC(=O)C(F)OC(F)(F)F)CC1 C12(CNC(C(C)N(C)C)=O)COCCN1C(=O)CN(C(c1cccnc1)=O)C2 C1(Nc2cc(OC)nc(C(F)(F)F)n2)CC2CCC(C1)N2CC1CCC2CC2C1 N1(C(C2(CC)CCCC2)=O)CC2(CC(NC(=O)C(c3ccccc3F)C)CO2)C1 N1(C(Cc2c(C)non2)=O)CCC(NC(=O)C(C)OC(C)(C)C)C1C(C)(C)C C(=O)(CC(C)(C)CN(C)C)NC1CCCN(C(C23CCC(OCC)C2C3)=O)C1 N1(C(C2(C)CC2)=O)CCCC2(C1)CN(C(=O)CC1CCC(=O)N1)C2.CCOC CC(CN(C1CC1)CNC(c1ccc(CO)s1)=O)C(=O)NC1(c2ccccc2)CC1 C1(=CC(=O)N(C(C(=O)N(CC(F)Cl)C)C2CC2)C)CCOCC1 C1(C(N2C(CC(C)C)CC(O)C2)=O)C2C3CCC(C3)C12 c12cc(cc(F)c1)CC(=O)OCCC1CCCCN1C2=O.C1(OC)CC(O)C1 c1(-c2c(OC)cnc(F)c2)c[nH]c2ncc(C(=O)Nc3cnn(CCO)c3)cc12 c1(OC)ccncc1NC(C1C2CN(Cc3nccn3C)CC12)=O CC1CN(C(=O)CCC(=O)N(C)C)CC1NC(=O)CC1CC=CCC1 C1(NC(=O)CCN2N=CCC2=O)CC2(NC(c3cc(F)ccc3F)=O)COC1C2 N1(C(c2cc(C(C)=O)c(C)o2)=O)CC2(CCC2NC(=O)C#CC(=O)N(C)C)C1 c1(C(N2CC(OC(CC)CSC)C2)=O)nc(NC(c2ccccc2)C)ncc1Br c1(CC(N2CC(NC(C(CC)C)=O)(COC)C2)=O)c(C)n[nH]c1C c1(C(CC(C)(C)CC(=O)O)=O)nc(C2CCc3c(Br)cccc32)no1 N1(C(c2csc(-c3ccccn3)n2)=O)CCC(NC(C2(F)CC2)=O)C(F)(F)CC1 C(=O)(CC(C)(C)O)N(C1CCN(C(C2(c3cncnc3)CCCC2)=O)C1)CCC c1(C(C)C)nccc(=NCC2CN(C(C3CCCC4(CC4)C3)=O)CCC2(F)F)[nH]1 c1(CNC(c2cncs2)=O)cccc(CNC(C2CCCCC2C(F)F)=O)c1 C1(C(N2CC(CNC(C3(c4ncccn4)CC3)=O)OCC2)=O)CC2(CC(=O)N2)C1 c1(C(=O)NCC(C2CCC2)NC(C(CC)(C)O)=O)ccc2c(c1)N(C)CC2 CCCCC(CC)C(=O)N(C1CCN(C(=O)CC2CCCO2)CC1)CCO N1(C(C(C(CC)O)C)=O)CCC2CCC(C1)N2C(c1ccc(NC=O)cc1)=O C=C(Cl)C(C)(C)C(=O)N1CCN(C(=O)C(C)CCC2CC2)C(c2cn[nH]c2)C1 N1(C(CN2C(C)CCCC2)=O)CCCC(F)(CNC(C2CCSC2)=O)CC1 C12(CNC(C3CC=CC3)=O)CCCC1CCN2C(c1ccc(C(N)=O)nc1)=O O=C(CN1C(=O)Cc2ccccc21)NC1CCCCCC1N c1(C(=O)NCCCC(C)NC(c2cc(Cl)ccc2Br)=O)ccnc2ccnn12 C1(C(N2CC(N(C(=O)CCC(=O)c3cccs3)C)C2)=O)Cc2ccccc2C1 C=CC(C)(C)CC(=O)N1CC2(CNC(=O)C(SC)SC)CCC1C2 C(CCN(C(=O)C(O)CC1CCCC1)C)(C(C)C)NC(c1cc(C)on1)=O c1(C(N2CCC(NC(c3nn(C)c(CO)c3)=O)C(F)C2)=O)ccc(N)c(F)c1F CCC(C)C(=O)NCC1(NC(=O)C(C)(C)n2cnnn2)CCC1 N1(C(C=C(CC)C)=O)CCC(C)(C)C(CNC(=O)C(O)P(C)(C)=O)C1 C1(C(N2CC(CCNC(c3cnc(C)nc3C)=O)C2)=O)CCc2cnc(C)n2C1 N1(C(CC2C(NC(c3ccc(C)cc3F)=O)CC2O)=O)CCCCC(F)(F)C1 N1(C(CC(C)SC)=O)CCN(C(=O)C=Cc2cocn2)CC1CCO C(=O)(C(O)C1=CCCCC1)N1CCCC(N(C(C(=O)NCC(F)F)=O)CCO)C1 C(=O)(C(C)(C)C(C)NC(=O)COC1CCCOC1)N1CC(C)OCC1 c1(N2CC(CCNC(c3conc3C)=O)(OC)C2)nc2cc(Br)cnc2s1 CCC(CC)CCCC(=O)NC1CCN(C(=O)CNC(=O)C(CC)CC)C1CC n1(C(C)C)cnc(C(=O)NCCCN(C(=O)C=CC2CCCO2)C)c1 Cc1csc(C(=O)NC2CCN(CCNC(=O)CCC3CCC(C)O3)CC2)c1C CCC(C)(C)C(O)C(=O)NCC1CCCCN1C(=O)COCCCC(C)C CCCCC(C(=O)Nc1cc(CC)cnc1O)NC(C1CCNC1=O)=O CC1CCC(CC(=O)NCCCNC(c2nc[nH]c2C(C)(C)C)=O)C1 C#CCCCCCCC(=O)N(CC(C)O)CCNC(=O)CCC(C)N(C)C C1(CC(=O)NC2CC(CNC(C(C)(C)n3cccn3)=O)C2)CCCCC12CC2 C1(C(=O)NC2CC(COC)C2)C=CCCN1C(C1C(C(C)=O)C1(C)C)=O C1(CNC(C2(CC=C)CCOC2)=O)CN(C(=O)CCc2nncs2)CC(C)(C)C1 Cc1cc2c[nH]nc2cc1C(N1CCC(F)(CNC(=O)CC2CCCCO2)C1)=O N1(C(C(C=CCCC)O)=O)CCCN(C(c2cn(C)nc2COC)=O)CC1C c1(N2CC(=C(C)CNC(=O)Cc3sc(O)nc3O)C2)cc(O)nc(O)n1 c1(CNC(C(=O)NC(c2ccccc2F)C)=O)ccnc(C#N)c1 C1(CC(N2CCC3C(NC(CC(CN(C)C)(C)C)=O)C32)=O)CCCC2(CCC2)O1 Cn1nc(CNC(C2CCSC2)=O)c2c1CCN(C(=O)CC1C=CCC1)C2 Cn1ncc(C(N2C3CCC2CN(C(=O)CCF)C3)=O)c1S(C)(=O)=O c1(C(N2CC(OC)C(NC(c3coc4c3CSC4)=O)C2)=O)cccn2nnnc12 c1(CC)cc(C(=O)NCC(C)CNC(=O)C(C)n2ccnc2)c(C)nn1 c1(C(=O)NCCN(C(=O)CC2CCCCC2)C(C)C)ccc(=O)n(CCO)c1 C=CC1(O)CCN(C(C2CCCN2C(=O)C(F)C(C)(F)F)=O)C1 N1(C(c2ccc(Cl)c(OC)c2N)=O)CCCN(C(=O)C(C2CC2)OC)CC1C c1(CN(C)C(c2cn(CCC#N)nn2)=O)nc2c(s1)CCCC2(C)C Cc1ccc(C(N2CCCC(Cc3nccn3C(C)(C)C)CC2)=O)c(Br)c1 C(CC(C)(F)F)(C(=O)O)NC(=O)NC(CCC=C(C)C)C C1(CN(C(=O)CC23COC(C)(C2)C3)C)C2Cc3c(Cl)cccc3C12 C1(OC)CN(C(=O)C(N2CC3(CC3)CC2CC(=O)O)=O)CCC1CC(=O)O c1(OC)cc(N2CCN(C)CC2)ccc1NC(=O)NC1COC2(COC2)C1 c1(C(=O)NCCC(C(=O)NC2C3COCC23)OC)cc(C)cc(C)n1 C1(C(=O)NCC2N(C(C(F)=C(C)C)=O)C3C(C2)C3)CCOCC12CCC2 C1(C(=O)Nc2ccnc(OC)n2)(CNCc2ccc(COC)cc2)CC(C)(C)C1 CC1CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CCC1NC(=O)CC(=O)NC1CC1 C(C(CC(=O)NOCCCCCC1CC1)C1CCC1)NC(=O)CC1CCCCC1 N1(CCNC(CC2(CNC(C(C)n3ccnn3)=O)CC2)=O)CCNC1=O C1(CNC(c2c(COC)cco2)=O)CCCN(C(C23CCCC2C3)=O)C1 N1(C(COc2cccc(CC)c2)=O)CC2CC(F)(F)C2C1 CC(C)(CCCNC(C1CN2CCC1(C)CC2)=O)C(=O)NOCc1cccnc1 C1(C(N2C(CNC(=O)CCCn3cccn3)COCC2)=O)CN2CCCN1CC2 C(=O)(C1=COCCO1)NC(CNC(c1c(C)csc1)=O)C(C)C C(=O)(CCCS(C)(=O)=O)NCC1C(NC(c2n[nH]c(C)c2Cl)=O)C1 C(C(O)CN=c1[nH]cnc2c([N+](=O)[O-])cccc12)NC(C(CC)F)=O C(C(CC(C)C)NC(c1cc(=O)n(C)o1)=O)NC(c1ccc(CCC)s1)=O c1(SC(C)C(=O)NC(C)(CNC(C2CC(F)(F)C2)=O)CO)nnnn1C1CC1 Cc1cc(=O)c(C(=O)NC2CC3(NC(=O)COC4(C)CCC4)COC2C3)cn1C C(=O)(C1CCCc2sc(C)nc21)N1CC2CC(NC(COCC#C)=O)C2C1 C(=O)(CCCCCCC1CC1)NC1CCC(N(C(=O)CNS(N)(=O)=O)C)C1 C1(C(=O)NCC2(C(F)F)CCN(C(=O)C3=CCOC3)C2)CC2OC1C1CC21 Cc1ccc(C)c(C(N2CC3CC(NC(=O)CCCc4ccccc4)C3C2)=O)c1 C1(NC(CCC(=C)C)=O)CC(O)CN(C(=O)COc2ccc(C)cc2F)C1 c1(C(=O)NC(C(=O)NCC2(CCOCC)CC2)c2cccs2)n[nH]cc1C c1(CC(C)C)ccc(CC(=O)NCC(O)CNC(C2CNC(=O)N2)=O)cc1 C1(C(N2C(CCC)COCC2)=O)CC2CC1CC2NC(=O)CC1CCC(=O)C1 C1(NC(c2ncc(CC)s2)=O)CCC2CC1CN2C(C1CC2CCC1C2)=O C1(n2cc(-c3n(C)ccn3)nn2)CCN(C(=O)C(=O)NC2CCC3CC3C2)CC1 c1(C(=O)NCC(CC)(C)NC(c2ccoc2CN)=O)cc(N(C)C)cc(Cl)c1 C(C)(N=c1[nH]nc(C2CC2)o1)C1N(C(c2cc(CC)on2)=O)CCCC1 c1(C(=O)NC(C2CCCN2C(c2n[nH]cc2Br)=O)C)ncc(F)cc1N N1(CCN(C2CCN(C3CCC3)C2)C(CC)=O)CCCOCC1.C(=O)OC C=CCCCCCCC(=O)N1CC(NC(=O)CCC(C)(C)F)C2CC12 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CC(C)CN(C(=O)CN2CCSCC2)C1 C12(C(N3C(C(=O)NC)CCC3)=O)CC(CN(C(c3nonc3C)=O)C1)C2 Cc1nc2cccc(C(=O)NCC3(C)CCCC3NC(=O)Cc3ccoc3)c2[nH]1 CC(C)CC(C(=O)N1CC2CC(C1)N(C(=O)CC1CCC(O)C1)C2)C(C)C c1(OC)ccc(-n2nc(-c3occc3C)nc2C(C)(C2CC2)C2CC2)cc1 C(=O)(C(C)(C)CC(=O)NCC(C)NC(=O)C(F)C(CC)CC)OCC Cc1cc(C(N2CC(CC(=O)NCC(C)(O)C3CC3)C3(CC3)C2)=O)cc(C#N)c1 N1(C(COCC(=O)OC)=O)CCC(NC(C2CCC(C3CC3)O2)=O)C(C)(C)C1 c1(C(=O)NC2CCN(C(c3cn(C)[nH]c3=N)=O)CC2O)cc(=O)n2ccsc2n1 CC1(C)C(=O)NCC1NC(C1(CNC(c2c(I)ccnc2F)=O)CC1)=O N1(C(C2(N(C(=O)Cc3cccnc3O)C)CC2)=O)CC(C)(C)CCC1CO C(=O)(N1OC2CCC1C2)C12CN(C(c3nc(OCC)oc3)=O)C(C1)CO2 N1(C(C2OCCN(C)C2=O)=O)CCC(C)(C)C(NC(c2cc(C(N)=O)cs2)=O)C1 Cc1nc(C(=O)NC2(C(=O)N(CCCN3CCCC3)C)CC(O)C2)sc1C C(=O)(C(C(C(C)C)C(C)C)NC(c1cc(O)ccc1F)=O)OC Cc1ccc2c(C(=O)NCC(C)N(C)C(c3cnc(C(N)=O)s3)=O)csc2c1 c1(CC(N2CC(C(C)NC(c3cnn(C4CCC4)n3)=O)C2)=O)c(Cl)cncc1Cl c1(CN2C(C3(O)CN(C(c4cccc(Cl)c4)=O)C3)CCC2)c(Cl)ccc(F)c1F CCC(C)(C)CCCC(=O)NC1CCCCC1NC(c1cncc(Cl)c1Cl)=O N1(C(C2(F)CCN(C(CCN(C)CCO)=O)C2)=O)C2C=CCC1CCC2 c1(C(=O)NCC2(F)CN(C(C=CC(=O)OCC)=O)C2)sc2ccc(C)cc2c1C C1(CC(=O)N(C(C)(C)C(=O)O)C)CCCN(C(C2CC2Cl)=O)C1 c1(C(=O)NCC2N(C(C(CCC)C)=O)CCCCC2)cccc2c1NC(=O)CO2 C#CC1(C(=O)N(CC(C)CO)C)CN(C(=O)C(F)CCC)C1 c1(CC)cc(F)c(C(=O)NC2CC(NC(=O)C3=CC(C)(C)C3)C2)c(F)c1 c1(C(=O)OC)c[nH]ccc1=NC1CC(NC(=O)CC2CCCO2)C1.C1CO1 c1(CNC(C(CN(C(C2(CC=C)CC2)=O)C)C)=O)ccnc(OC)c1 CC(C(=O)NC1CC(N(C(=O)Cc2ccc(Br)c(O)c2)C)C1)S(C)(=O)=O N1(C(=O)NC(c2c(Cl)cccc2Cl)C)CCC2(CCCNC2=O)CC1 c1(C(=O)NCC(C)N(C(C2(COC)CCCC2)=O)C)ccc2c(c1)NC(=O)C2=O C1(CCCC)CN(C(=O)C(C)C2CCCC2)CCN1C(c1ncc(N)cc1C)=O N1(C(C2CCC3CC23)C(=O)NCCC2(C)CC2)CC(C(N)=O)C(c2ccccc2)C1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CCC(NC(Cc2nc(C)c(C)s2)=O)C1 CCC(CC(F)F)C(=O)NC1(C)CC(NC(=O)CCCSc2ccc(Cl)cc2)C1 c1(OC)ccc(C(=O)NCCN(C)C(C2CC(SC)C2)=O)s1 c1(NC)ccc(S(=N)(=O)C(F)(F)F)cc1.CC1CCC2CN1C(=O)N2 c1(C(=O)OC)ccc(NCC2CCc3ncnn32)c(C#N)n1 CC(C)C(C(=O)NC1CCCC1C(C)C)NC(=O)CC1CCOC1(C)C c1(CC)ncnc(N2CC(NCc3ncc(F)cc3F)CC(C)C2)c1F c1(CC)ccc(NC(=O)NC(CC)C(C)O)c(Br)c1 O=C1CCC(CC(=O)NC23CC2CN(C(c2cccc(OCC4CC4)c2)=O)C3)CN1 c1(C(=O)Nc2c(NC(c3cnc(C(N)=O)nc3)=O)nccn2)cc(F)ccc1Cl C1(CNC(CCCSC)=O)COCCN1C(C1CC1c1occc1Br)=O c1(C(N)=O)ccnc(NCC(N2CC(O)(CCNC(C3C=CCC3)=O)C2)=O)c1 C1(CC)CN(C(=O)CC2CCC(C)(O)CC2)CCN1C(=O)C=C(Cl)Cl CCCC(CCC)C(=O)NC(CNC(C1C(C(C)=O)C1(C)C)=O)C1CC1 c1(OC2CCN(S(=O)(=O)Cc3ccon3)C2)cc2c(cc1F)NC(=O)CC2 Cc1ccc(C(=O)NCCCC(C)(C)NC(c2cnc(O)cc2C)=O)c(N)c1 c1(C(N2CCC(CCC(=O)N(C(C(C)SC)C)C)CC2)=O)coc2ccccc12 CC1CN(C(c2ccncn2)=O)CCCN1C(=O)CC1CCC(C)O1 C12(C(=O)NCCNC(C34COCC3C4)=O)CCC(C(F)(F)F)(CC1)CC2 C1(NC(=O)CCC2CC2)CCCC2CN(C(=O)C(F)(F)C3CCCC3)CC12 N1(C(CCSCC)=O)CCC(C)N(C(=O)CC(C)C(F)F)CC1 C1(C(=O)NCc2ncc(CC)[nH]2)CN(C)CCN1C(c1cc2n(n1)CCO2)=O C1(C(C)NC(=O)Cn2ncnn2)CCCCN1C(=O)COc1ccsc1 CCC(C(=O)NCC1(O)CN(C(=O)C(c2ccccc2)O)C1)n1ccnc1 N1(C(CCCOCCC)=O)CCC(C)C(CC(=O)NC(c2nccs2)(C)C)C1 c1(C(=O)NC(C)(C)C)ccnc2ccc(F)nc12.C1CC(=O)NCCCC(=O)N1C N1(C(C(C)C2CCOC2)=O)CC(C2(NC(c3cnc(O)c(Cl)c3)=O)CC2)C1 CCC(C(=O)NCc1ccncc1)NC(=O)CC(C)n1cccn1 C12(CC)CCCN(C1)C(=O)c1c(cccc1)C(=O)N2.c1(CC)c[nH]c(C(N)=O)c1 C(=O)(C(F)(F)Cc1ccccc1)NCC(CNC(Cc1cn(C)nc1)=O)O C1(CC)CN(C(C2CCSC2)=O)CC1C(=O)NCCC(=O)NCC(C)C CC1CCN(C(=O)Cn2cnnc2O)CC1NC(C1(CS(N)(=O)=O)COC1)=O C1(CC)CCCC1C(=O)NC1CC(CC(=O)N(CCN2CC=CC2)C2CC2)C1 c1(C(=O)NCC(CC)NC(c2nnn(-c3ccccc3)c2C)=O)cncc(N)n1 CC(C(=O)NCCOC1CCN(C(c2cscc2Cl)=O)C1)P(C)(C)=O C#Cc1ccc(C(N2CC(C(=O)NC3CC(N(C)C)C3)C3(CC3)C2)=O)cc1C CC1CC(C)(C(=O)NC2CC(CNC(C3(c4ccc(Cl)nc4)CC3)=O)C2)CCO1 C1(CC)(CC)CCN(C(C23CC2CCN3C(c2ccc(C)o2)=O)=O)CC1 c1(COC)ccc(NC(C2C(C)CCN2C(=O)CC(C)c2ccco2)=O)cn1 C(N=c1[nH]c(=NC2CN(CC(F)F)C2)[nH]c2c1COC2)c1c(C)cc(C)cc1C c1(C(N2CCC(NC(c3c(C)n[nH]c3C)=O)C2C)=O)cn(C)ccc1=O C1(CN(C)O)CCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(CCC)cc(C(=O)N(CC)CC2CCN2C(=O)Cn2nnnc2C(C)C)nn1C c1(C(N(CCNC(C(C)=C2CCCC2)=O)C)=O)cc(-c2cccnc2)on1 CN1C(=O)CSC1=CC(=O)N1CC(CO)(NC(c2cc3c(s2)CCCC3)=O)C1 C1(CNC(c2c(N(C)C)nccc2)=O)CC(N=c2[nH]ccn3ccnc23)C1 C(CC(=O)Nc1cc(Cl)cnc1O)(C(C)C)NC(C1(C)ON=C(C)C1)=O N1(C(C(CC)F)=O)CC(C)CN(C(C2CCC(C)(O)CC2)=O)CC1C c1(C(N2C(CNC(CSCCC)=O)CCC(C)C2)=O)c(F)ccc2ccoc12 c1(OC)cc(CN2CCCCC2C(=O)NCc2cc(O)cc(O)c2)cc(F)c1O c12ccc(cn1)S(=O)(=O)NC1CCN2CC1.N1(S(C)(=O)=O)CC(O)C1 C(CCCN=c1[nH]c(=NC2CCC3CC2CO3)c2c(ncn2C)[nH]1)OC c1(C(CO)N(C(C2C(C(=O)OC)C2)=O)CC2CC2)ccnn1C.C1C(=O)N1 C1(NC(C=CC(C)(C)C)=O)C2CC(CN(C(=O)Cc3sc(O)nc3O)C2)C1CO N1(C(c2c(C(C)C)ccs2)=O)CCCC(NC(=O)C(F)(F)c2cncs2)CC1 N1(C(C(C(CC)CC)F)=O)CC2(CCCN(C(=O)CCc3ncc(C)[nH]3)C2)C1 Cc1cccc2c1OCC2C(=O)N1CC(CCNC(c2ccc(F)cc2O)=O)C1 c1(C(=O)NC2CCN(C(c3cccc(CC)c3O)=O)CC2)cc(C)c(C)cc1N c1(C(N(CCNC(c2c(C)nn(C)c2N)=O)CC)=O)cn(C)c(=O)nc1O c1(C(=O)NC2C(CC)N(C(c3scnc3C)=O)CC2)cc2cccc(C)c2s1 c1(C(N(C2C(O)CCN(C(C(C=C)O)=O)C2)C)=O)ccn2nnnc2c1 C1(C(=O)NCC(C)(C)OCC(=O)N(C(CCSC)C)C)CCCCC1O c1(CNC(C(C)(C)C2CCCN2C(=O)COCC2CCC2)=O)ccncc1F CC#CC1CN(C(c2ccc(-c3ccc(Br)cc3)s2)=O)C1 CC1(C)CC(NC(C23CCC(C2)C3(C)C)=O)CCN(C(=O)CCc2nc[nH]n2)C1 c1(C(N2C(CCNC(C3COC(=O)N3)=O)CC(OC)C2)=O)cc2n(n1)CCO2 c1(OC)cc(C)c(CC(=O)NCC(C)NC(=O)CC2CC(C)C2)c(C)c1 Cc1cc(Br)c(C(N2CC(O)C(O)C2)C(N2CCC(CN(C3CC3)C)CC2)=O)s1 CC1C(NC(C2CCNC(=O)C2)=O)C(C)CCN1C(c1cccn2nnnc12)=O N1(C(=O)CON)CC(F)(F)CC1CO.c1(CC)ccccc1O CCC(CC(=O)NCCCCN(C(=O)C(C)NC(=O)OC(C)(C)C)C)C(C)(C)C N1(C(C(C)C)=O)CCC2(CC2)CC1C(=O)NC1CC2(C)CCC1CC2 c1(C(N(CC(C)(C)C(=O)NCCNC(=O)C(C)(C)C)C)=O)cc(C#N)ccc1N C1(C(N2CC(C=C)C2)=O)(NC(=O)CC(C)(C)OC)CCN(C)C1 c1(CC)ccc(C(=O)NC2CCN(C(=O)C(F)CC3CC3)CC2O)c(Cl)c1 c1(C(N2CCC(CCNC(C=C(C)C)=O)C2)=O)ccn2cnc(C)c2c1 C1(CCC(=O)NC2(COC)CCOC2)CCN(C(C2(C)CCOC2C)=O)CC1 C(=O)(C1=CC(C)CC1)NC(=O)NC1CN(CCCNC)C(=O)C1 N1(Cc2ccc(SC)c(Br)c2)C2CCCC1CC1(C2)NC(=O)NC1=O C1(NC(CS(=O)(=O)NCC)=O)CCCC12CCN(C(c1cc(C)c(N)cn1)=O)C2 Cc1cc(C#N)cc(C)c1C(=O)NC1CC(NC(c2cnsc2C)=O)C12CCC2 Cc1nc(NCC(c2ccccn2)(F)F)nc(Cl)c1Br C1(N(C(COC(C)C)=O)C)CCC(CNC(=O)CC23CCC(CC2)C3)CC1 c1(NC(C2C3CN(C(C(C)OCC#C)=O)CC2C3)=O)ccc2nc(C)[nH]c2c1 c1(CN(C(CS(Cc2cccc(C)c2)(=O)=O)=O)C(C)(C)C)oc2ccccc2c1C c1(C(N(CC(CC)NC(C2(COC)CC2(F)F)=O)CC)=O)nnc(S)n1C C(=O)(CC1CCc2ccccc21)NCC(CN(C(C1=C(C)CCC1)=O)C)C C1(NC(C(C2CCN(C(C3(CO)CC(C)(C)C3)=O)C2)F)=O)CCC2CC2CC1 CC(C)CC(C)C(=O)NCC1CN(C(c2c(F)cncc2Cl)=O)CCN1C c1(CCC(=O)NC(CC(C)NC(COC)=O)C)cccc(N(C)C)c1 CC(C)C(C)(C)C(=O)NC1CC2CC(NC(=O)C(N3CCC(O)CC3)C)C1C2 CC(CS(C)(=O)=O)C(=O)N1CCCC(CO)(NC(c2cc(=N)[nH]c(Cl)n2)=O)C1 c1(CN2CC(C)N(c3ccn4nccc4n3)CC2)c(Br)ccc(F)c1F C(C)(C(=O)NC1CC(CC(=O)N(C)CC2(C#N)CC2)C1)SCC=C c1(CC(N2CC(Cn3cc(C(C)(C)O)nn3)OC(C)C2)=O)nsc2ccccc12 N1(C(CCCCC)=O)CCCC12CN(C(c1nc(C)ncc1Br)=O)C2 C12(CNC(C(COC)NC(C)=O)=O)CCC(C1)N(C(=O)COC(F)F)C2 Cc1coc(C=CC(=O)N(C2CCCN(C(=O)C(C)n3cccc3)C2)CCO)n1 C(C)(CCC(=O)NC1(COC)CN(C(C2CCCN(C(C)C)C2)=O)C1)OCC c1(OC)c(C)nc(C2CC2)[nH]c1=NCCC1(Cc2cccc(F)c2)CC1 C#Cc1ccccc1CC(=O)NC1CCN(C(C2CC(OC)C(OC)C2)=O)CC1 C(=O)(CC(C)C(F)F)N1C(CCNC(=O)CNC(c2ccsc2)=O)CC(OC)C1 C1(NC(=O)Cc2cnccn2)CN(C(=O)CCc2ccc[nH]2)CC2(CCC2)C1 N1(C(c2cc(OC)n[nH]2)=O)C2CCC1CC(C(=O)NCC1CC3(CCC3)C1)C2 Cc1sc(-c2ccccc2SC(C)(C)C)nc1C(=O)NC1(C)CCC1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCCC(C)(NC(c2c(CC)ocn2)=O)C1 c1(C(=O)NC(CC(=O)NCc2ccc(C)s2)(C)C)cc(F)cnc1O N1(C(C2(C#C)CCC2)=O)CC(NC(=O)C(c2c(C)noc2C)(C)C)CC(C)C1 C1(CN(C(C(C2CC(F)(F)C2)OC)=O)C)CCN(C(=O)C(C)CC2CC2)C1 N1(C(C(C)OCC2CCC2)=O)CCCC(c2n[nH]c(CNC(=O)C(C)(C)C)n2)C1 C#Cc1ccc(NC(C2COCCN2Cc2cnc(OCC)cn2)=O)cc1 N1(C(c2ccncc2F)=O)CCC2(CCN(C(=O)CC3CCCCC34CC4)C2)C1 C(CCCCC)(C(=O)NCC(C)C)c1cccc(-c2ccc(CC)cc2)c1 N#CC1(C(=O)NCC2CCCC2NC(=O)CCc2ccccn2)CCSCC1 C1(NC(COC(C)=O)=O)CC(CNC(C2CC2(C)C(F)F)=O)C1 C#CCCC(O)C(=O)NCC1(CNS(C)(=O)=O)CN(C(=O)Cc2ccccc2F)C1 N1(C(C(C)c2ccsn2)=O)CCCC12CCN(C(=O)CS(=O)(=O)CCO)C2 C1(NC(=O)CO)CCN(C(=O)Cc2cscn2)C12CCC2 C1(CC)C(=O)NCCCN1C(C1CC(C)(C)CCN1C(=O)C(C)OC(C)(C)C)=O c1(C(N2CC(OCCF)C2)=O)cc(CNC(=O)C=CC(F)F)[nH]n1 C(=O)(C(C)(C)CCCNC(=O)CCCF)N1CCCC(COC)C1 O=C1OC2C(CNC(c3ccccc3)CN3CCCC3=O)C2O1 C(=O)(C1CCc2nccn21)NC1(CC)CCN(C(=O)CCC(=O)NC)C1 N1(C(c2c(C)noc2C)=O)CC2(CC(NC(=O)CN3CCCCCC3=O)CO2)C1 c1(C(=O)NCCCCC(C)NC(=O)C2=CCSC2)cn(C)ccc1=O C1(NC(C2(CNC(C(CC)C)=O)CCCC2)=O)CC2CC(O)C1C2 c1(N2CCC(CCn3cccn3)C2)[nH]c(=NCC2CC3CCC2CC3)nc2sccc12 c1(SCCNC(C2N(C(COC(C)=O)=O)CC=C2)=O)nc2ccccc2cc1C C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC2CN(C(c3c(C)cncc3)=O)C(C1)C2 N1(C(C(CC)=CC)=O)CCC(NC(C2CCCCC2(C)C)=O)C(C)C1 c1(C(=O)NCC2CN(C(C(C)CN3CCCCC3)=O)C2)cnc2c(F)cccn12 Cc1ocnc1-c1cn(CCCCCNC(=O)Cc2csc(Cl)n2)nn1 c1(OC)nc(C(=O)NCC2OCCC2C(=O)N(C)CCOCC(F)F)co1 C1(CN(C(C(C2CCC2)OC)=O)C2CC2)CCCN1C(=O)CNS(N)(=O)=O c1(C(=O)NC(C)(CNC(=O)C(O)CC2CCCC2)C2CC2)cccc2ccoc12 c1(C(CC)(C)C)ccc(N2CC(C(=O)NCc3ccc(C)nn3)C2)cc1 N1(C(C2CC(OCC)C2)=O)CC2(CCN(C(c3nnsc3C)=O)CC2)CC1C C1(C(NOCCOCCOC)=O)CCC(O)CN1C(c1cncc(C)c1)=O c1(CN2CC(NS(C)(=O)=O)C2)ccc(NC(C2CC3CC3C2)=O)cc1 C(CCCCC(=O)NCCOCCCNC(=O)C(C)n1cccn1)OC Cc1coc(C)c1C(=O)N(CCCCN(C)C(c1cnc[nH]c1=N)=O)C c1(CN2CCCC(Cc3nnc(C)n3C)CC2)cc2c(nc1O)CCSC2 CS(=O)c1ccc(-c2cnc(NC(c3cccnc3Br)=O)c(O)c2)cc1 C1(NC(C(C)C(F)F)=O)CC2(CCN(C(C3CCCN(CC(F)F)C3)=O)CC2)C1 c1(OC)ncc(Br)c(N2CCC(C)C2CNC(c2ccc(C)c(O)n2)=O)n1 c1(C(N2CCCC(NC(N3C(C)CCCC3C)=O)C2)=O)c(F)cc(F)cc1Cl C(CC(C)C)(C(=O)N1CCC(N(C(=O)C=C(C)c2ccsc2)C)C1)NC(C)=O CN1CC(C(=O)N(CCCCCC(=O)NC2CC(O)C(O)C2)C)CCC1=O C(CCC(C)C)(C(=O)NC1(CNC(C2(C)CC2C)=O)CCOCC1)NC(C)=O C(=O)(C(C(=O)NCCc1ocnc1CNC(c1cncn1C)=O)C(C)C)OCC CC1CC(CNC(c2cccs2)=O)CN1C(=O)C(C)Cn1ccnc1 C1(CNC(=O)CSC2CC2)CN(C(C2CC2Cc2ccccc2)=O)CCO1 C(=O)(C1CCOc2ccc(Cl)cc21)NCC1CC(NC(=O)C#CC2CC2)C1 C(=O)(C(O)C1=CCCCC1)NCC1C(C(=O)NC2CC(C)(C)OC2=O)C1(C)C CC1=C(C(=O)NC2CC(F)CN(C(=O)C(F)(F)C(F)F)C2)CCCO1 C(=O)(CCCS(C)(=O)=O)NC(CNC(C(CCC)=CCC)=O)C(C)C(C)C Cc1cccc(F)c1CC(=O)NC(C)C(CO)NC(c1cc(O)ccc1Br)=O N1(C(C2(CC=C)CC2)=O)CCC(C(C)CNC(c2cc(CC)sn2)=O)CC1 c1(C(N2CCN(C(CCC=C(C)C)=O)CC2)=O)c(C#N)ncn1C c1(NC2C(C(=O)Nc3cncc(OC)c3)CCCC2)ncc2c(ccn2C)n1 C(=O)(CCC(C)(F)F)NCC(C)CNC(=O)COCc1ccccc1Cl C1(CNC(C)=O)CN(C(C23CC(C2)C(C)O3)=O)CC1C C1(CC(=O)NC(CNC(C=CC(C)C)=O)(C)C(C)C)CC(=O)NC(=O)C1 Cc1ccc2c(C(=O)N(CC(C)NC(C3CCC(C)O3)=O)C)ccnc2c1C c1(CC)ccc(C=CC(N2CCC(CNC(=O)CN3CCCC(CC)C3)C2)=O)o1 Cc1cc(O)cc(O)c1CN1CCC(C(N2CCC3(CCCO3)C2)=O)C1 N1(C(CS(CC)=O)=O)CCC(CO)(CNC(=O)CCc2cnn(C)c2C)CC1 N1(C(C2CCC(=C)CC2)=O)CC2CCN(C(c3cc(C)cnc3F)=O)CCC2C1 C1(O)(CNC(c2c(OC)csc2)=O)CCCN(C(=O)C=Cc2ccncc2)C1 c1(NCC(N2CC(N(C)C)C3(C2)CC3)=O)ccc(S(=O)(=O)N(C)C)cc1 C(C(CC(F)(F)F)NC(c1cc(Br)n[nH]1)=O)NC(c1cn(CCOC)nn1)=O N1(C(c2c(C)nc(-c3ccco3)[nH]2)=O)CC2CC1CCN2C(C1CCCC1C)=O O=C1CC2(CC(C(N3CC(OCCNC(c4ccc(O)nc4)=O)C3)=O)C2)N1 N1(C(C(C)OCCC=C)=O)CCC(NC(c2ccc(C#N)o2)=O)C1(C)C c1(OC)ccc(CN2CCC(F)(C(=O)Nc3nc(Br)ccc3C)C2)c(OC)c1 c1(C(=O)NC2C3CN(C(C(C)O)=O)CC2COC3)c(Cl)cc([N+](=O)[O-])cc1Cl N1(C(c2ccc(C#C)cn2)=O)CCC(NC(C23CCC(C)(C2)OC3)=O)C(C)(C)C1 N1(C(=O)C=CC=C2CCC2)CCOC(CNCc2ccc(Br)s2)C1 C(=O)(C(F)(F)C(O)C(C)C)N1CC2N(C(c3c(Cl)cc(C)nc3)=O)CC(C2)C1 c1(CC(N2C3C(NC(C(C(C)C)F)=O)C(CCC3)C2)=O)ccc(S(C)(=O)=O)cc1 C1(NC(c2c(C)occ2)=O)CC2(CCN(C(=O)C(C)(C)C)CC2)C1 c1(CC)noc(CCCC(=O)N(CC(O)CNC(=O)CCc2cn[nH]c2)C)n1 C1(N(C(c2ccc(O)cc2)C(F)(F)F)C(C2CC2F)=O)CCC12CCNCC2 C1(CNC(c2sc(F)cc2Cl)=O)CCN(C(=O)CCOC2CC2)CC1(F)F C1(C)(CCNC(c2c(CCC)n[nH]c2)=O)CCN(C(c2c[nH]c(C)n2)=O)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)N(C(C(=Cc1cn[nH]c1)C)=O)C1CC(N(C)C)C1 C1(C)(CC)C=C(C(=O)NCC2CCCN(C(=O)Cn3nccc3C#N)C2)C1 C1(C(N2CC3(CC(CNC(=O)CN4CCNC4=O)C3)C2)=O)Cc2ccccc2C1 C#CC1C(C(=O)N2CCC2)C1(C)C.c1(S)ccncc1.C(=O)(C(C)OCC1CC1)N c12cccc(n1)C(=O)NCCC1CCCN1C2=O.C1(C(N)=O)(C(N)=O)COC1 N1(C(Cc2cccc(OC(C)C)c2)=O)CCC(c2cn(CC(=O)O)nn2)CC1C Cn1c(C(=O)N(C2CCCCC2c2ccc(Cl)cc2)CC(=O)O)cnc1O N1(C(C(CC=C)c2ccccc2)=O)CCCC2(C1)CN(C(=O)C(C)CF)CCO2 N1(C(c2c(C)ccnc2)=O)CCC(CNC(=O)C(C)P(C)(C)=O)C(F)(F)C1 C1(CC(=O)NC(C)(C)CF)CC(O)CN1C(C1CC1(F)Cl)=O N1(C(c2cn(CC)nc2C)=O)CC2=C(C1)CN(C(c1ccnc(C(C)C)c1)=O)C2 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCCN(C(CC(C)(C)SC)=O)CC1C Cc1ncc2n1CCC(C(=O)NC1CCC(CNC(=O)C=CC(C)(C)C)C1)C2 C1(CNC(COCc2n[nH]c(=N)s2)=O)CCCCN1C(C1CCSC1)=O c1(CC)nc(C)[nH]c1C(=O)NCCN(C(=O)C=Cc1scnc1C)C1CC1 N1(C(c2ccc[n+]([O-])c2)=O)CCN(C(c2ccccc2Br)=O)C(C2CCC2)C1 N1(C(C(C)N(C(c2c(OC)scc2)=O)C2CC2)=O)CCC(N=[N+]=[N-])CC1 N1(C(C(SC)SC)=O)CCC2(CC2C(=O)N(C)Cc2cncs2)C1 C1(CCOC)(NC(=O)CCC(C)OC)CCN(C(=O)CSc2ccccn2)C1 C1(C(=O)NC(C2CCCC2)CC)C2CCCC2N1C(=O)C(C)n1cccn1 c1(-c2cc(SC)cc(C)c2)ccc(C(=O)NCc2c[nH]nc2C)c2[nH]ccc12 Cc1cc(C(N2CCCC2C#N)C(=O)NC2CCC2)c2c(c1)CCC2 N1(C(CN(CCC#C)C)=O)CCCC(N(CCO)C(C2CNC(=O)C2)=O)C1 Cc1ccc(C(=O)NCCCOCCNC(c2ccc(F)cn2)=O)c(C)c1Br c1(CC)nc(C(N2CCCC(CNC(C3CCC(N(C)C)CC3)=O)C2)=O)c(N)s1 c1(SC)c(C(=O)NCCCOCCNC(c2n[nH]cc2C2CCC2)=O)cnn1C N1(C(c2cc(F)cc(Cl)c2)=O)CCCC12CCN(C(C1(CO)CCCCC1)=O)C2 C1(C(=O)NCC2(CO)CC(C)C2)CCCN(C(c2cc(O)nc(O)n2)=O)CC1 C1(C)(OC)CCSCC1.C1(C(c2nnnn2C2CCCCC2)(C)NCCC)CC=CCC1 c1(C(=O)NC2C(F)CCN(C(C3C(C)(C)NC(=O)C3)=O)C2)cnc2[nH]cnc2c1 C1(C)(C(=O)NC(CNC(C2C(CC)CC2)=O)C2CC2)CCOC(C)C1 C12(NC(c3ccc(CO)c(F)c3)=O)CCCC1CN(C(=O)CCc1nncs1)C2 C12CC(=NO1)C(=O)NC2.Cc1cnn(CCC(=O)NCCSC(C)(C)C)c1 C#Cc1ccc(C(N2CC3(CC(NC(=O)C(C)OCCC=C)CO3)C2)=O)c(C)c1 c1(C(CC)=O)ccc(NC(=O)CNC2C(C)C2(C)C)cc1 CCCCCC(C)CC(=O)NCC1(C)CCN(C(=O)C(C)CCOC)C1 c1(C(N2CC(C)N(C(C3CCSC3)=O)CC2)=O)ccnc2ccncc12 C1(C)(CC)CCCN(C(c2ccc(C(F)F)cc2C)=O)CC1 C1(NC(C2C(C)(CC)C2)=O)CN(C(c2ccc(CO)c(Cl)c2)=O)CCC1C N1(C(C2CC(NC(C3C(CC)OCC3)=O)C2)=O)CCC(C2CCC2)CC1 N1(C(=O)NCC2(NC(N)=O)CC2)CCCSCC1C1CC1.C(F)(F)F C(CCF)(C(=O)NC(C)CCC1CCCC1)NC(c1c(C)occ1)=O Cc1ccc(CC(=O)N(C)CC2(NC(C3CC3C(C)(F)F)=O)CC2)o1 N1(C(CCCCC=CC)=O)CCN(C(=O)C=CCN(C)CC)CC(C)(F)C1 c1(C(=O)NCCCCCn2cc(-c3ccsc3)nn2)ncc2cc(Cl)ccn12 c1(C(N2CCC(C(C)NC(c3cccc(Cl)c3O)=O)C2)=O)c(F)cc(F)cc1Cl C(c1ccccc1F)=CC(N1CCN(CC2CC(O)C2)C2CC12)=O CN1C(=O)CC(NC(C2(NC(=O)CC(C)(F)F)CCCC2)=O)C1=O N1(C(c2c(C)nc(S)s2)=O)CCCC2(CCN(Cc3ncc(Cl)cc3F)C2)C1 c1(C(=O)NC(CN(C(C(C)CSc2ccccc2)=O)C)C)ncc([N+](=O)[O-])n1C C1(O)(CC(N2CC(NC(C(C)OCC)=O)C(OC)C2)=O)CCCCCC1 Cc1c(C(N2CC(O)CC2CNC(c2nnn(C)c2C)=O)=O)nc2sccn12 C(=O)(C(C(C)(C)C)N1CCNC1=O)NCCC(C)NC(C1CC(C#N)C1)=O C=CCCCC(C(=O)NCc1nc(=O)o[nH]1)NC(C1CCC2(CCC2)O1)=O c1(SC)c(C)cccc1Br.C12CCN(CC1)C(=O)CCCc1nnc2s1 c1(C(=O)NCC(CN(C)C(c2nc(C(N)=O)cs2)=O)O)cc2ccsc2n1C N1(C(CC(CCC)NC(C2(c3ccccc3)CC2)=O)=O)CCn2ncc(C)c2C1 C1(C(=O)NCCN(C(c2coc(O)n2)=O)Cc2ccccc2)CCOCC12CCC2 c1(CC)c(NC(=O)C(C2CCN(C(C3(C(=O)N(C)C)CC3)=O)C2)C)cnn1CC c1(C(N(C2CCN(C(c3ncn(-c4ccccc4)n3)=O)C2)C)=O)sccc1C#N CC1(C)C(CNC(=O)COC(C)(C)CNC(C2CC2[N+](=O)[O-])=O)C1(F)F C1(C(C(=O)NCCN(C(CC)=O)C2CC2)C)CCCCN1C N1(C(CC(C(C)C)O)=O)CC2CCC1(CNC(c1ccc3c(c1)OCO3)=O)CC2 C1(OC)CCC(N2CCN(C(=O)C(C(C)C)N3CCCCC3)CC2)CC1 Cc1cccc(Br)c1C(C(=O)Nc1ccc(O)c(Cl)c1)NC(=O)CSC1CCC1 CC(CCCNC(c1ccc(CN2CCCCC2)o1)=O)NC(=O)CSc1cccs1 c1(C(=O)NC(C2CCN(C(C3(C)CCC(=O)C3)=O)C2)C)cc(O)ncn1 N1(C(c2cnc(C(C)(C)C)s2)C(=O)NCCC)CC(OC)CC(OC)C1 CC1CCCCC1(CNC(C1C(C)(C)OC1(C)C)=O)NC(=O)Cn1cc(Cl)cn1 N1(C(c2ccc(Cl)nc2C)C(=O)NCCCOC)Cc2ccccc2C1 c1(C(C)NC(N2CCCC(c3cc(F)c(Cl)cc3Cl)C2)=O)cc(Cl)c(F)c(Cl)c1 CCCCC(C(=O)N1CCCC(F)(F)C1)NC(C1CCN(CC)CC1)=O C(C)(C)(C(C)CC(=O)NCC1(C2CC2)CCCO1)NC(C1C=C(C)CS1)=O C1(NC(C=C(C)Cl)=O)CCCC(CNC(=O)CCC2CCC(=O)N2)C1 c1(C(=O)NC(C)C(CO)NC(c2ccccc2)=O)cc2cc(Br)ccc2[nH]1 C(C(CNC(=O)Cc1ccccn1)C(F)(F)F)NC(=O)CC1COCCO1 C#Cc1cccc(CNC(c2ccccc2)C(F)F)c1 N1(C(C(C)CC#N)=O)C2CCC1CN(C(c1ccc(C3CC3)cc1)=O)C2 C(=O)(C(=O)C(CC)OC(=O)CCc1ccc(C(F)(F)F)cc1)OCC C(=O)(C(C)(C)C(=O)NC(CSC)CC(C)C)OC.C12(C)CCN(C1)C2=O C1(NC(C(F)=C(C=CC)CC)=O)C2CC3CN(C(=O)CC4CC4)C1C3C2 c1(SC)ncc(C(=O)N(CC(C)NC(C2CCC3(C2)N=N3)=O)C)c(O)n1 C1(NC(C(C)NC(N)=O)=O)CN(C(=O)C#CC2CCCOC2)C2CCCCC12 N1(C(CCC=C)=O)CCCC2CN(C(c3ccc(O)cc3CC)=O)CCC12 CC1CCC(CC(=O)NC2(C(=O)NCCC(C)(C)O)CC2)O1 c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)OC)=O)ccc2nccn2c1 C1(N(C(c2cc(CN(C)C)on2)=O)C)CCCN(C(=O)C(F)n2cccn2)C1 C1(NC(C(CC=C)C)=O)CN(C(c2ccc(F)c(C(=O)C3CC3)c2)=O)CC1(C)C CS(=O)(=NC(=O)C1CCC1(F)F)c1cnn2c1CN(C(C1CCC(=O)N1)=O)CC2 C#CCCC(C(=O)NCc1nc(CCC)no1)NC(c1cn(C2CC2)nn1)=O C(C)(CC(N)=O)N(C(C=CC(C)NC(=O)Cc1cn(C)cn1)=O)C CC1CCOCC1C(N1CCN(C)CC1)=O.C(=O)(CN(CC=O)C)NCCO N1(C(c2cnc(CC)[nH]2)=O)CCC(NC(c2cnn(CCF)c2)=O)CC1C c1(C(N2CCN(C(CCC(C)OC)=O)CC2CO)=O)cc(C)nc2ccccc12 CN1CCCC(C(N2CCCCC2CNC(c2cn(C)nc2C(F)(F)F)=O)=O)C1 C1(NC(CC2(C)CC2(F)F)=O)CC2CC(C1)N(C(C=CC(=O)NC1CC1)=O)C2 c1(C2(C(N3C4CN(C(=O)C5CC5)C(C4)C3)=O)CC2)c(Cl)cccc1Cl CCC(C)C(C(=O)NC(c1cnn(CC)c1)C)NC(=O)CC1(OC)CCC1 c1(C(=O)NCCCCC(C)NC(c2c(C)nc[nH]2)=O)ccc(F)cc1Cl N1(C(C(C(C)C)NC(C)=O)=O)CCC(C(=O)NCCCCl)C(O)C1 c1(C(C)=O)ccc(S(=O)(=O)N2CC3C(C2)N3C(=O)CCn2nc(C)cc2C)cc1 N1(CCCC)CCOCC1C(=O)NC(CNC(C1CCCC1O)=O)C(C)(C)C C(CCC(=O)NC1CC1C(=O)N(C)CC1(C)CCCO1)OC(C)=O C(CC(C)(C)NC(=O)C(C)C1CC1c1ccccc1)NC(C(C1CCC1)OCC)=O c1(NC(C23CC(COCC)(C2)C3)=O)ccc(Sc2cc(C)no2)c(C)c1 C1(C(N(C2CCN(C(C)C)C2)C)=O)CCN(C(=O)CCc2ccn(C)n2)CCO1 C(CCC(C)C)(C(=O)N1OC2CCC1C2)NC(CCCC1C(C)=C1)=O N1(C(CCc2ccc(C)s2)=O)CC(C)CN(C(c2ncn(C(C)C)n2)=O)C(C)C1 C1(CC)C2CCOCC12.c1(C2c3nnnn3-n3nnnc3CN2)cc(Br)cn1C c1(C(=O)NC2C(NC(C(CCCOC)C)=O)C2)cc(C)nc2ncnn12 Nc1c(Cl)ccc(C(N2CC3(C2)CN(C(c2ccco2)=O)C3)=O)c1Cl C(=O)(C(F)C(F)(F)F)N(C(C(F)(F)CO)C1CC1)C C1(CN(C(Cc2c(C)non2)=O)C)CC(F)CN1C(=O)Cn1ccsc1=N N1(C(CNC(CNC(C2C(C)C2)=O)=O)=O)CC2(CCN2C)C1 C(=O)(CCS(C)(=O)=O)N(CCN(C(=O)CCSCC)C(=O)CSC(F)(F)F)CC.CC C1(N(C(c2ccccc2)=O)CC)COCCN1C(c1cnc(-c2ccoc2)s1)=O c1(C(=O)NC23CC(CNC(CSCC=C)=O)(C2)C3)ccc(N)c(C)c1C c1(C(N2CC(CNC(c3cc(C(C)=O)on3)=O)C2)=O)cc(C)n(C(C)C)n1 c1(C(N2CC(O)(CCNC(C3N(C)C(=O)CC3)=O)C2)=O)cc2c[nH]nc2s1 CCCCC(C(=O)NC1CC(NC(=O)Cn2nnc(C(C)(C)C)n2)C(O)C1)OC c1(C(=O)OC)cc(N2CC(CO)(NC(=O)C(C)OCC(C)C)C2)ncn1 c1(OC)ccc(F)c(C(N2CC(CC(N)=O)CCC2C)C(=O)NC(C)C)c1F Cc1ccc(Cl)c(C(N2CCC(C)(NC(=O)COC3CCCC3)C2)=O)c1O C12CN(CC(C)O1)C2=O.c1(COC(=O)OC(C)(C)C)ccc(C(C)(C)C#N)cc1 C(=O)(CC(C)Sc1nncn1C)NC(C1(O)CN(Cc2ccccc2)C1)C N1(C(C(C(C)(C)C)NC(CSCCCC)=O)=O)CC2(C1)CN(C)CCO2 C(=O)(CC(O)C(C)C)NC(C(=O)NCC(C#C)CC1CC1)CCC1CC1 N1(C(CCCC)=O)CCCC2CN(C(C3CC4CCC(C3)O4)=O)CCC12 CC(C(=O)N(C)CC1(O)CN(C(C2CCC(F)(F)C2)=O)C1)C(F)(F)F N1(C(C2CC3CCC2C3)=O)CCC(CNC(C2(CO)CCCO2)=O)C12CC2 C(CCCCCN(C)C(C1CN(C)CCO1)=O)NC(CNC(C)=O)=O O=C(CS(=O)(=O)C1CCCC1)NC1CCCC1C(=O)NCCN1CCOCC1 C(CCC(=O)NCCN(C(=O)C(C)(F)c1ccccc1)CCC)=CCC=C C1(CNC(C=CCC)=O)CC2CCC1N(C(c1csc(-c3ncc[nH]3)n1)=O)C2 C1(CCC(=O)NCCC(C)NC(C2(n3nccn3)CC2)=O)CCCN1C CCCCCC(CC)C(=O)N1CCC2C(NC(=O)CCC(=O)OC(C)(C)C)C2C1 c1(C(N2CCC(C)(CNC(c3cnc(C)[nH]3)=O)C2)=O)cnc(Cl)c(C)c1 N1(C(c2ccc(C3CC3C)o2)C(=O)NCCC)CC2(C)CCC2(C)C1 C1(C)(C(N2CCC(OCCNC(CCSCC(C)C)=O)CC2)=O)CCCS1(=O)=O C1(NC(c2nc(CC)sc2)=O)CCN(C(=O)C=C(C)C(C)(C)C)CC1O C1(C(N(c2ccsc2C)CC)=O)CCCC(NC(C)=O)C1 c1(CCC)nc(-c2coc(-c3csc(C)n3)c2)n(C2CCSCC2)n1 Cn1cc(C(N)=O)c(-n2cc(-c3ccc(OC(F)F)cc3)nn2)n1.O(NC=O)CC CCCC(O)C(=O)N1CC(CO)(NC(c2cc(Br)c(Br)s2)=O)C1 C(c1ccc(Cl)cc1)=CC(C)NCC(c1noc(CO)n1)OC N(C1c2ccccc2CC1NC(c1cnn(CC)c1C)=O)C(C=CC)=O c1(C(N2CCC(CCCCCOCC)CC2)=O)cccc2ncnn12.C1C(=O)N1 C(c1ccc(F)c(F)c1)=C(C(=O)NC1CC(CNC(C(CCCOC)C)=O)C1)C C(C(O)CC(=O)NCCC1COCCN1C(c1ccc(CCF)cc1)=O)N(C)C C1(C(=O)NC(CCC=C(C)C)C)CC(O)CN1C(=O)CC1CNC(=O)O1 C1(OC)CN(C(=O)CC(C)c2ccncc2)CC1NC(C1(C)CC(C#N)C1)=O c1(C(=O)NC2C(CNC(C(C)OCOC)=O)C2)cc(F)ccc1C.C(C)(C)(C)S CC(O)C(C(=O)N(CCNC(=O)CN1CCOCC1)Cc1ccccc1)N(C)C c1(C(=O)NC(c2ccccc2)CNC(C(C=C=C)C)=O)cc2cccn2c(O)n1 c1(CCC(=O)NCCCN(C(C(C(CC)O)C)=O)C2CC2)cc(F)c(F)c(F)c1 CC1C2CCCCC2CN1C(C1CC(NCc2nccs2)C1)=O C(=O)(CC(C)(C)CCOC)NC1(CC)CCN(C(=O)C(F)C(C)(F)F)C1 c1(C(=O)NCC(CCCC)NC(C2(F)CCS(=O)(=O)C2)=O)ccc(F)c(O)c1 Cc1c(C(=O)NCCOCCOCCNC(=O)C(C)(Cl)Cl)ccc2n[nH]cc12 C(=O)(C1SCc2cccnc21)NCC1CCN(C(C2C(C)(C)C2)=O)CC1 c1(SCC(=O)NCCC(C)NC(c2cncnc2)=O)ccccc1Br c1(OC)ccc(Cl)cc1C(N1CCCC1CNC(=O)C(CC(C)C)C1CCC1)=O n1(CCC)nc(-c2cccc(C(F)F)c2)nc1-c1ccnc(Br)c1 C(C(C)(C)CN(C(=O)Cc1ccns1)C1CC1)NC(C(C)OCCOCC)=O C1(C(=O)NCCOCC(=O)N(C)CC2CCCC2(C)C)CCOCC1(C)C N1(C(C2(C)C(C)(C)C2)=O)CC=C(C(=O)NC2CC23CCCCC3)C1 N1(C(c2cc(C)oc2)=O)CC(C2CCCN(C(=O)Cc3c(C)cccc3C)C2)C1 C1(NC(CSCC#C)=O)CCSC12CN(C(=O)Cn1cnc(C(F)(F)F)n1)C2 N1(C(C2=C(C)CC2)=O)CCN(C(=O)C(CCC2CC2)NC=O)C(C(C)C)C1 N1(C(C(C2CC2)OC)=O)CCC(CNC(c2cn(-c3cccnc3)nn2)=O)C1 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NCC1C(NC(=O)C=Cc2cc[nH]n2)CC1 N1(C(C=C(C)Cl)=O)CC(N(C)C(c2ccc(C(N)=O)cn2)=O)C(F)C1 C1(NC(C2(NC(C)=O)CC2)=O)CCC(NC(c2cc(C3CC3)ccn2)=O)CC1 CC1=C(C(=O)NCC2CCCC(CNC(=O)Cc3ccc(CO)cc3)C2)CCO1 CCC1CC(=O)N(C)C1.c1(CC2CCCN2C(=O)C2=CSCS2)ccccc1C c1(CNCCCNC)cc(C)ccc1SCCC(=O)OC CP(C)(=O)CCC(=O)NCC(O)CNC(C1CC(Cc2ccccc2)C1)=O Cc1ccnc(C(=O)NCC2(O)CN(C(=O)CCCNC(c3cccs3)=O)C2)n1 CCC(CC)(CC)C(=O)NC(c1ccccc1)CNC(=O)C(C)OCCN(C)C c1(C(=O)NC(C)CCNC(c2ccc(CCF)cc2)=O)ccc(Br)c(O)c1 c1(C(N2CCC(CNC(C(CC)(F)F)=O)C(C)C2)=O)cc2c(C)ccc(F)c2o1 C=C(C)C1OCCC1C(=O)NCC1(C)CCCN(C(=O)CSC)C1 Cc1c(C(=O)NC2CC(CNC(C3(C(C)C)CC3)=O)C(O)C2)[nH]c2c1CCCC2 C1(NC(CC2C(C)(C)C2(C)C)=O)CN(C(=O)CC2OCCCO2)CC2(CCC2)C1 C(C(C(=O)NC1(CF)CCC1)NC(C1CCOCC1)=O)OCC.C1CC1 C(C)(CCC(=O)N1CCC(NC(c2cccnc2S)=O)C1C)OC C1(N(C(C(n2ncc(C)c2)C)=O)C)CCC(C(N)=O)CC1.C1(O)(CC)CN(C=O)C1 C12(C(N)=O)CCCC1(C(N1CC(NC(=O)CCCC3CC3)CC1CO)=O)C2 C1(O)(CNC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(c2cnc(O)o2)=O)CC1 C12(CNC(c3cc(Cl)no3)=O)CCC(CC1)CN2C(=O)C=Cc1cccnc1 c1(C(=O)NCCC(CNC(c2cnc3c(c2)NCC3)=O)O)c(F)ccc(F)c1Cl N1(C(c2c(COC)n(C)nc2)=O)CC2(CCN(C(c3coc(CO)n3)=O)CC2)C1 c1(OC)c(C(N2CCC(CNC(=O)C(C)(C)OC(C)=O)C(C)C2)=O)ccnc1F Cc1ccc(Br)cc1CCC(=O)N(CCCCNC(c1c(C)ncn1O)=O)C Cc1ccnc(C)c1C(=O)NC1CCCC1CNC(c1cccc(C)c1C)=O c1(C(N(C)CC2CN(C(C(C)OCC#C)=O)C2)=O)[nH]c2ccc(OC)cc2c1C CCC(CC(=O)N(C)CCN(C(=O)C(=Cc1ccccn1)C)C(C)C)C(F)F Cc1ccc(Br)cc1C(N1C2CCC1C(NC(c1ccnnc1C)=O)C2)=O N1(C(C(C)N(C(C)=O)C)=O)CCN(C(=O)Cc2nnc(C)s2)CC1c1cn[nH]c1 N1(C(C=CCN(C)C(c2ncccc2F)=O)=O)CCSC2CCC12 C1(CCN(C)C(C2CC(O)C(F)C2)=O)CCN(C(C2(C3(C)CC3)CC2)=O)CC1 c1(C(=O)NC(C(C(C)C)NC(CCc2cnc(C)s2)=O)C)cc2cnccc2o1 C1(NC(C(C)C2CC2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC2(CCC2)C1 N1(CCC(=O)NCCC2CCN(C(C(C)C(C)(F)F)=O)C2)Cc2ccccc2C1 CON(CCC(=O)NCC12CCCCC1C2)C(=O)c1cc(C)no1 C1(CNC(C(Cn2cncn2)NC(=O)CCc2cnn[nH]2)=O)NC(=O)NC1=O N1(C(CN(C(CCN(C)CCO)=O)C)=O)CCCC(C#N)C1 C(CC(C)C)(C(=O)NCCCSCCO)OC.c12n[nH]cc1C(=O)N2 C1(CC(=O)Nc2cnn(C3CCCC3)c2)CCCC1NC(C1(O)CCOC1)=O CCCCC(CC)CC(=O)NCC(C(=O)NCc1cccnc1F)N(C)C c1(NC(C2CCN(C(C(C(CC)O)C)=O)CC2)C)ncc(C#N)cc1Cl c1(N2CC(CC)SC(C)C2)nccc(=NCc2ncccc2Br)[nH]1 c1(OC)ccc2c(c1)CCCN2S(=O)(=O)CC12CCC(C1)C(=O)N2 C1(CC#C)(C(=O)NC(CNC(=O)C=CCN(C)CC)CC)CCOC1 C1(NC(CCC(=O)NCC)=O)COC2CN(C(=O)CCS(C)(=O)=O)CC12 C1(C(C)C)(C(=O)NC2COC(=O)C2)CCN(C(c2cc(C3CC3)no2)=O)C1 CCCC(C)(CC)C(=O)N1C2CC1CN(C(=O)Cc1ccc(C)s1)C2 c1(C2C(C(N3CCC(CC(C)NC(C)=O)CC3)=O)C2)cc(Cl)cc(Br)c1 n1(CC)cc(NC(C(C2CCN(C(C3OCCC3C)=O)C2)OC)=O)cn1 c1(C(=O)NC(c2csnn2)C)coc(C(C)NC(C2(O)CCSC2)=O)n1 C1(CC(C)O)CCCN(CC(=O)Nc2ccc(-c3ccc(Br)cc3)n2C)C1 C1(C(=O)NCCc2ncn(C)c2)(NC(=O)CC23CCC(CC2)C3)CCC(C)(C)C1 N(C1CCCc2ccccc21)C(C1(C)CCN(c2ncncc2F)CC1)=O N1(C(C(CC)Oc2ccccc2Cl)=O)CCC(O)(C(=O)NC(C2CCC2)C)CC1 C1(C(=O)NCC(CNC(c2n(C)c(O)nc2)=O)(C)F)CCCC(C(N)=O)CC1 C1(COC)CN(C(=O)C(C2(O)CCCC2)F)CCN1C(=O)CN(C1CCCC1)C N1(C(c2ccc(CC)c(CC)c2)=O)CC2CC1CN(C(=O)CC1CCCO1)C2 c1(CC(=O)NC2CC(C)CN(C(c3c[nH]c(=O)cn3)=O)C2)cc2ccccc2o1 C1(O)(C(C)C)CCCN(C(=O)CC2(NC(=O)COCCF)CCC2)C1 c1(NCCCCSC)ccc(S(=O)(=O)N2CC=C(c3cccs3)CC2)c(Br)c1 C12CC(CC1O)C(=O)N2.N1(C(N)=O)CC(C(N2CCC2C(=O)NC2CC2)=O)C1 c1(-c2ccc(C(=O)NC(CN(C(=O)CC3CC(F)C3)CC)C)o2)ccc(O)cc1 C(CCCCCC(=O)NC1CCCCC1NC(C12CC(O)C1C2)=O)SC C1(NC(C(CC)N(C)C)=O)CCC(N(C)C(C2(C)CCCOC2)=O)CC1 c1(OC)nc(O)ccc1NC(=O)COC1CCN(C(=O)C=Cc2cccnc2)C1 N1(C(C2CC2C2CC2)=O)CC2OCC(NC(C34CCCN(CC3)C4)=O)C2C1 CC1CCN(C(c2cnccn2)=O)CC1CNC(=O)Cc1ccc(Cl)cc1 Cc1cc2c(Br)ccc(C(N3CCCC4C3CCN4C(C3CC3C)=O)=O)c2o1 CCCC(O)C(=O)N1CCN(CC2CN(C(c3nncn3C3CC3)=O)C2)CC1 Cc1cc(N)c(C(=O)NC2(C)CN(C(C3CCCSC3C)=O)C2)cc1C CCC(C)(CO)C(=O)NCC(C)(C)NC(C1C(C2CC2)C1(F)F)=O C(C(CC)(CC)C(=O)N(CC(c1nn[nH]n1)C)C)NC(C1C(C(=O)OC)C1)=O C1(c2nnnn2CCSC)(Nc2c(SCCC)cc(F)cc2)CCC(C)(O)CC1 N1(C(C(c2ccccc2Cl)C)=O)CCN(C(c2cc(Cl)cn2C)=O)C(CO)C1 c1(C(N2CC(C)(C(N3CC(C(C)(C)C)C3)=O)C2)=O)ccc(N)cc1 Cn1cccc(C(=O)NC2C3CN(C(=O)CCc4cnn[nH]4)CC23)c1=O Cn1nc(C(=O)O)c(-c2cn(CCNC3CCCN(c4nccs4)C3)nn2)c1Cl C=CCCC(C(=O)NC(C)CCOCC)NC(c1cc(O)ccc1C)=O c1(OC)ccc(F)cc1-c1nc(C(O)CC(C)O)n(-c2ccc(Br)nc2)n1 C1(NC(C(C)NC(CC)(C)C)=O)CN(C(c2nc(C)oc2C)=O)CC1C N1(C(=O)CCc2ccsc2)CCC(F)(CNC(C2(C3CC3)CCOCC2)=O)CC1 N1(C(C(C=C)(F)F)=O)CC(CNC(=O)CC2CCN(C)C2=O)OC2(CCC2)C1 C(=O)(C(CC)C(C)C)NCC(=C)CCNC(c1cccc(OC(F)(F)F)n1)=O N1(C(CC2CC(=O)OC2)=O)CCN(C(c2ccc(CO)nc2)=O)C2CCCC12 c1(C(=O)NCC2N(C(CC(CC)CC)=O)CC(O)C2)oc(S(N)(=O)=O)cc1C N1(C(C2N(C(C3N(C)CC(F)C3)=O)CCOC2)=O)CCC(CO)=C(F)C1 C(CCN(C)C)(C(=O)N1CCCC1C1CCOC1)NC(C1CC(C)C1)=O C(=O)(C(CC)CC(F)F)NCCN(CCC)C(c1oc(COC)cc1C)=O C(=O)(CCC(=O)C(C)(C)C)NCC(C(C)C)C(=O)NC1(C)CCOCC1 CCCCCC(=O)N1CCOC(C(C)NC(c2n[nH]cc2CC(=O)OC)=O)C1 C1(C(N(C2CCN(C(=O)Cc3ccc(C)nc3)CC2)CC)=O)CCCOCC1 Cc1ccn2cc(C(=O)NC(C)CCCNC(=O)CN3CCN(C)CC3)nc2c1 N1(C(C2N(C)CC(F)C2)=O)CCC(C)(C)C1CNC(=O)NC1(CCN=[N+]=[N-])CC1 c1(C(=O)NC2(CC=C)CCN(C(C3(C)CCC3)=O)C2)cc2cccc(C)c2s1 C1(CC(=O)NC(C(=O)NCCC(=O)NC(N)=O)C2CCOC2)COCC(C)O1 C1(OC)CN(C(c2cn(C)c(-c3ccccn3)n2)=O)CC1F c1(C(CCCN(c2ccccc2)C(C)CCO)O)cncc(F)c1 CC(CN(C)C)CCC(=O)N1CCC(OCC(N2CCC(F)(F)CC2)=O)C1 CCCC(CCCNC(=O)C1=NOCC1)NC(c1c(C)[nH][nH]c1=N)=O C1(CN(C)C(C2(C)CC(F)(F)C2)=O)CN(C(=O)C(C)(C)C2CCCC2)CCO1 c1(C(=O)O)nc2ccccn2n1.Cc1ccc(OCc2noc(C)n2)cc1C N1(CC(=O)N(C(C(C)C)C)C2CC2)C2CCCC1CN(C(C1CCCN1C)=O)C2 c1(CC(=O)NCC2CC(C(=O)OC)C2)cc(Cl)ccc1Cl.C12CCCC1C(=O)N2 C1(NC(c2c(CC)cns2)=O)(CF)CCN(C(c2csc(Cl)c2Cl)=O)C1 N1(C(C2CC(C)NC(=O)C2)=O)CC2CCC(C1)N2C(=O)CCc1ccoc1 C1(C(N2CCN(C(C(C(C)O)C)=O)C(C)C2)=O)CCC(N=[N+]=[N-])CC1 C(=O)(CCC(C)C)NCC(CC=C)NC(=O)CNC(c1cccc(F)c1)=O C1(C(N(C)CC2CCC2)=O)CN(C(C2CC23CC3)=O)CC1C1CC1 C1(C(=O)NCC)N(C(C2CC(F)CN2C(=O)OC(C)(C)C)=O)CC1(C)C CC1CC(NC(c2cnc(C(C)(C)C)o2)=O)CN1C(=O)CN(C)C(N)=O c1(N2CC(NC(c3ccncc3F)=O)CC3(C2)CC3)nc(Cl)nc2c1CCOC2 CCC(CC)CCC(=O)N1CC2CCC2(CC(=O)NCc2csc(C)c2)C1 c1(OC)cccc(C(=O)NC2CCC(C)(NC(C)=O)C2)c1OC CCCCC(F)C(=O)N1CCC(NC(=O)C(C)OCC(C)C)CC1C c1(C(=O)NC2(C)CN(C(Cc3cn(C(C)C)nc3)=O)C2)c[nH]c2c(F)cccc12 Cc1cnc2n1C(C(=O)NC1CC1CNC(c1cn3ccsc3n1)=O)CCC2 N1(C(C(COC)O)=O)CCC2(CC1)CC2NC(c1ccc(-n2cccn2)cc1)=O c1(C(=O)NC2CC(N(C(C(CC=CC)C)=O)C)C2)cc2cccc(C)c2o1 C1(C(NOc2c(C(=O)NC3C(OCC)CCC3)ccnc2)=O)CC12CCCCC2 CCC(CC)CC(=O)N1CCC1C(=O)NC(C)CC(F)(F)F N1(C(c2cc(C)no2)C(=O)NCCCSCC)CCCCC1C1CCCO1 N1(C(C(N)Cc2ncccn2)=O)CC2C(C(F)(F)F)(C1)CS2(=O)=O c1(C(=O)NC2CN(C(=O)C=CC3CCC3)CC2F)ccc(F)c(C(F)(F)F)c1F C(=O)(CCCCN=[N+]=[N-])NC1C(NC(C(n2ccc(C)n2)C)=O)CCC1 c1(NCC2CCCCN(C)C2=O)cc(S(=O)(=O)NCc2ccon2)ccc1C#N C1(NC(c2nc(OCC)sn2)=O)CN(C(c2cc(C)c(C)s2)=O)C2(CCCC2)C1 c1(N(C)CC2CN(C(=O)CSC(F)F)C2)nc(-c2cncs2)nn1C c1(-c2cn(CCN(C(c3cccnn3)=O)CC)nn2)ccccc1OC1CCOC1 c1(C(N(C)CC2CCCN(C(C3CCNC3=O)=O)C2)=O)coc2c1CS(=O)(=O)C2 N1(C(CCn2ccc(C)n2)=O)CCCC(N(C(=O)CC2CCCC2O)C)C1 c1(C(=O)NCCN(CCOC)C(c2cnc(C(C)C)nc2)=O)cnccc1Cl N#Cc1cccc(NC(C2CCC3(CC3)N2C(C2CCOCC2)=O)=O)c1 c1(CC)[nH]c(C(=O)NCC2(NC(c3cncc(C(F)(F)F)c3)=O)CCC2)nc1Cl c1(C(=O)NC(C2CCCCN2C(=O)CCC(=O)N(C)C(C)C)C)cn(C)[nH]c1=N c1(C(=O)NC2CC(NC(C(C)(C)N3CCCC3)=O)C23CCC3)coc(S(C)(=O)=O)c1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1(C)CCCN(C(=O)CSCC#N)C1 Cc1cc(C)nc(CNC(C2(NC(C3CCCCCCC3)=O)CCCC2C)=O)n1 C(C(C)(O)C(F)F)NC(CCC1(NC(COCC#C)=O)CCC1)=O C(C(C(=O)NCC(CC)N(C)C)NC(=O)C(F)n1ccnc1)OCC Cn1cnc2cc(CC(=O)NC3C4CN(C(C5(O)CC5)=O)CC34)ccc12 Cc1nn(C)c(C)c1OCCNC(=O)NCc1cccc(-c2ccsc2)c1 c1(C(N2CCC(N(C(c3cn(C4COC4)nn3)=O)CC)C2)=O)cnc(Cl)n1C C(=O)(C1CCN(C(=O)C(C)Oc2ccccc2)c2ccc(OC)cc21)OC C1(OC)CC(NC(=O)C(C2CCCCCC2)O)CN(C(=O)CC(C)(C)OC)C1 C1(NC(c2ccc(CCC)cc2)=O)(CO)CCN(C(c2nccnc2C)=O)CC1 Nc1cc(C(=O)NC2CC2CNC(c2ccccc2C2CCC2)=O)ccc1Cl c1(C(=O)NCC2(F)CN(C(C(CC)SC)=O)C2)n[nH]c2ccc([N+](=O)[O-])cc12 CC(C)(C#N)CCC(=O)NCC=CC(=O)NCCC1CCC1CO C(CCCC(F)(F)F)NC(C(=O)NC(C)C)CCSC N1(C(c2occ(C)c2C)=O)CCC2CN(C(=O)C(c3ccc(F)c(Cl)c3)C)CC12 c1(CN(c2cccc(N(C)C)n2)C)cccc(OC(F)F)c1 c1(C(N(CCCNC(c2cccc(COC)c2)=O)C2CC2)=O)cc(C#N)[nH]c1C CC(C)(CC#N)C(=O)NC1CCC(Cn2cc(CC3CC(F)(F)C3)nn2)CC1 CCCCC(C(=O)NC(C)C(F)(F)F)NC(C1COCOC1)=O N1(Cc2ccncc2)CCc2sc(-c3cc(N4CCOCC4)cs3)cc2C1 c1(OC)cccc2scc(C(N3CC4(CCN(C(C5(O)CC5(C)C)=O)C4)C3)=O)c12 C(C(=O)NCCc1cncs1)(C1(O)CCC1)NC(CNC(C1C(C)C1)=O)=O C(=O)(C1CCCn2ccnc21)NC1CCCCN(C(c2ncn(CC)c2)=O)C1 C(=O)(C1=C(C)CC(C)(C)CC1)NCC1CC2(C(OC)(OC)CC2)C1 Cc1n[nH]c(C)c1CCC(N1CCC(C)C1CNC(c1cn(CCO)nn1)=O)=O O=S(=O)(c1ccccc1C(F)(F)F)CN1CCCCC1CC1CCCC1 C1(CNC(=O)C(O)C2CN(C(C3CC(F)(CF)C3)=O)C2)CCCC2CC12 N1(C(Cc2ccc(OC)cc2)=O)CCN(C(c2cnccc2C)=O)C(CCO)C1 C(CC(C)C)(C(=O)N(CCNC(c1ccccc1)=O)CCOCCO)OC.C(C)(C)N c1(C(=O)NCC(=O)NC(CNC(C(C)n2cncn2)=O)C)ccccc1 OC1CCCc2c(NCCCn3cccn3)ccnc21 Cc1ccc(CNC2CC(=O)N(C3CC3)C2)c(C)c1Br CCCC(C)(C)C(=O)NC1CCCC(NC(=O)CC2C=CS(=O)(=O)C2)C1 CC1CC(NC(=O)Cc2nc(C3CC3)cs2)CCN1C(c1cnn(C)n1)=O c1(C(=O)NCCCC2(NC(c3cccc(O)n3)=O)CC2)nc2ccccn2c1F N1(CC(=O)NCC(CNC(c2cc(C)on2)=O)OC)CCSCC1 c1(CC(=O)NCCN(C(c2cccnc2C(F)F)=O)CC)cc2ccccc2o1 C#Cc1ccccc1NC(C1CN(C(c2cccc(F)c2C)=O)CCO1)=O N1(N(C(C)CS(C)=O)C)CCC(=O)C(C)C1(C)C N(C1CC(C)(CO)Oc2ccccc21)C(C(N1CCCC(CC)(OC)C1)=O)=O c1(C(=O)NCC2(O)CCN(C(=O)COCC3CCOC3)C2)csc2nccn12 C1(C(=O)OCC)CC(=O)N(C)C1C(N1CCC1CNC(C1CC(C)CCO1)=O)=O c1(C(N2CC(NC(C3CC4(CC4)C3)=O)C3C2C3)=O)cc(O)ccc1Br C1(NC(Cc2ccc(OC)cc2)=O)CC2(NC(=O)CN3CCC3C)COC1C2 CCC(CC)C(C(=O)N(CC(=O)NC(C)COCC)CCOCCO)OC N1(C(c2cnco2)=O)CC2CCN(C(C3(C4CC4)CC3)=O)CC2C1 CC12CC1CCN2C(C1CCN(C(=O)C2=NOCC2)C1)=O C1(C)(CNC(CS(CC)=O)=O)CCC(NC(c2cscc2C(=O)OC)=O)CC1 N1(C(c2c(CC)cncc2)=O)CCC(NC(C23CCCC2C3(F)F)=O)C(F)C1 C(CCCCC(=O)NCC1CC(C)(C)CN1C(=O)CC(=O)NC1CC1)OC N1(C(C(COC)(F)F)=O)CCC(NC(c2cccn(C)c2=O)=O)C(CO)C1 C(C(F)C(=O)NC1CCC(CNC(c2ccn(C)c2)=O)C1)N(CC)CC Cc1cc(CC(=O)NC2CCC2CNC(C2(C)CC=CC2)=O)cc(F)c1 CC1CCN(C(=O)OC(C)(C)C)CC1C(=O)O.C123COC(C1)(C2)NC(=O)OC3 c1(N2CCC(NC(CN3CC(C)(C)C3)=O)C(F)C2)nc(Cl)nc2ccccc12 N1(C(c2ccc(CNC(CC(C=C)(C)C)=O)s2)=O)CCC(N=[N+]=[N-])CC1 CCC(C)C(O)C(=O)N1CCCCC1CNC(c1ccc(C)nc1Cl)=O N(C(=NCCC1(C)CC1)NCC1CCCS1)C(C)C1CC1 c1(CCC)cc(C(N2CCN(C(=O)C(C)N(C)C)CC2)=O)c(C)o1 C1(Nc2ncc(C(=O)OCC)s2)(NC(=O)C(=O)Nc2ncc[nH]2)CCCCC1C c1(CNC2C(C(N3CCC4CCCCC4C3)=O)C2)c(Cl)ccc([N+](=O)[O-])c1Cl C(C(C)C)(C(O)C(=O)NC(CC(C)C)C(=O)NCCc1csc(C)n1)OC N1(C(CCN(C)CC)=O)CCCC1CN(C)C(c1csc(SC)n1)=O N1(C(C2N(CC)CCC2)=O)CCCC2(CCN(C(C3C4CCCOC34)=O)CC2)C1 C1(Cl)(CNC(=O)NCC(c2ccccc2Br)O)CC12CCC2 c1(C(=O)NCCCN(C(C(C(C)SC)O)=O)C2CC2)ccc2nnc(S)n2c1 CCC(C#N)C(=O)N(CCCNC(c1cnn(CCO)c1C(C)C)=O)C(C)C c1(C(=O)NC(c2cc(Br)co2)c2nnnn2CC2CCCO2)cc(Cl)cnc1O N1(C(C=CC=CC)=O)CCN(C(=O)CC(O)Cc2ccccc2)C(CCO)C1 c1(C(C)(C)C)nc(CNC(C2C=CCN2C(c2cncnc2)=O)=O)cs1 N1(C(C(C)N2CCCC2)=O)CC(C)C(C)(C(=O)NOCc2nc[nH]n2)C1 Cc1cc(N)cnc1C(=O)NCCC1CCCCN1C(=O)CC1CC1(C)C CCCCC(C)C(=O)N(CC(C)(C)C(=O)NCC1CCN(C)C(=O)C1)C C(CN=c1[nH]c(=NCCN2CCC(C)C2)[nH]c2cc(OCC)ccc12)C1(SC)CC1 C1(C(=O)NCC(C(C)C)NC(c2cnc(C(C)=O)s2)=O)CC2CCCC(C1)C2 c1(C(=O)NCC2CCC(NC(=O)Cc3c[nH]nc3O)C2)c[nH]cc(Cl)c1=O C(CN=c1nc2sccc2c[nH]1)C1CCN(C(=O)NC2CCCCC2O)C1 C1(NC(c2c(C)ccnc2)=O)CCN(C(c2cc(Br)n(C)c2)=O)C(C2CC2)C1 c1(CC)nc(=N)[nH]cc1C(N1CCCCC1CCN(C(=O)C=CC(C)(C)C)CC)=O Cc1ccc(C(=O)NCC2C3CC2N(C(c2cncc(C4CC4)c2)=O)C3)c(C)c1 c1(C(N2CCC(C#C)(O)C2)=O)n[nH]c2c1CN(C(=O)C=CC)C2 CC1COCCC1C(=O)NCCCN(C)C(c1cnc(C(C)(C)C)[nH]1)=O c1(C(N(CC(O)CNC(C2CC3CCCCC23)=O)C)=O)cc(Cl)c([N+](=O)[O-])[nH]1 N1(CC(N2CCC(C(N3CCOC4CC34)=O)C2)=O)C(=O)CCCC1=O C(=O)(CC(C(C)C)C(C)C)NCCC1(O)CCN(C(c2[nH]cc(CC)c2)=O)C1 c1(C(=O)NCC2C(C)CCN2C(c2cc(C#N)c[nH]2)=O)cncc2c1CCC2 c1(C(=O)OCC(N2CCCC(C(=O)OCC)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 Cc1cnc2n1CCCC2C(=O)N1CC(NC(=O)C(C)Oc2cccc(F)c2)C1 C1(C2CCN(C(C34CC3C4)=O)C2)(NC(c2cc(C(F)(F)F)n[nH]2)=O)CC1 N1(C(C(N2C(=O)CCC2=O)CC)=O)CCC(O)(CN(C(=O)CC2CC2)C)C1 C1(NC(c2ccc(OC(F)F)cc2)C)CCCCN(CC2CCC(C)(C)OC2)C1 C=CC(C)(CC)C(=O)N1CC(NC(C2CSC2)=O)C1 C1(CC=C)(NC(=O)CCc2cnn(C)c2)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 C(=O)(CC1C(=O)Nc2ccccc21)NC1CN(C(Cn2c(C)ncc2[N+](=O)[O-])=O)C1 c1(CC)cccc(C(=O)NC(C)C(C)C(=O)N(C)Cc2cn(C)nc2C)c1 c12cc(C)ccc1OC1(CCC1)CC(=O)N(C)C2.c1(COC)cn(C(C)C)nn1 C1(C(=O)NCc2c(C(=O)NC3(C)CSC3)scc2)CCCCC1CO c1(OC)ccc(C(N2CC3(C(N4CCCC4C)=O)CC2CO3)=O)cc1OC(F)F C1(C(N2CC(C)(C(C)C)OCC2)=O)CC(C)(C)CCN1C(=O)C1=C(C#N)CCC1 c1(CNC2CCCC(P(C)(C)=O)C2)cc(Br)cc2c1OCCC2 C(=O)(C1=NOC(CNC(C2CC(CC3CC3)C2)=O)C1)NC(C#CC#C)(C)C c1(C2CN(C3CCC(NC(c4nc(OCC)sn4)=O)CC3)C2)cc(F)cc(Cl)c1O Cc1cncc2cc(C(=O)NCC(C)(O)CNC(C3CCSC3)=O)sc12 CC1CCN(Cc2cc3ccsc3[nH]2)CC1c1cccs1 C#CCC(C)(C)C(=O)N(C)CCOCCC(=O)NCC(F)Cl C#CCC(C(=O)N1CCC(C(C)C(=O)N(C)C(c2ccccc2)C)CC1)C1CC1 c1(OC)ccc(CN2CCC2C(=O)NCCCCn2cc(CCO)nn2)cc1C N1(C(CC2C(C)CCO2)=O)CC(NC(=O)C2=CCCCO2)C2CCCCC12 C(=O)(C(C)(CO)NC(c1ccnc(CO)c1)=O)N(CC(c1ccccc1)O)C N1(C(COCC=C)=O)CC2CC1CN(C(c1cn(C)nc1C(C)C)=O)C2 C1(C(=O)NCc2c(C)cncc2)CC12CCN(C(c1cccnc1)=O)CC2 c1(C(N2CCC(C(C)(C)C)(CNC(=O)CC3CCC3)C2)=O)cc2cccnc2s1 C1(CCC)(CO)CCN(C(=O)C(C2(O)CN(C(C3CCSC3)=O)C2)F)C1 c1(C(C(C(C2CCCC2)N)=O)=O)ccnn1C1CC1.C(CNC(=O)C1CC1)N c1(C(N(C(C)CNC(=O)C(O)CC2CCOCC2)C)=O)cc(N)ccc1O C12(NC(C(C)N(C)C)=O)CC(CN1C(=O)CCCC1CC1)C2.C1(C2CC2)CN1 c1(C(=O)NCC2N(C(c3cn(C)c(Br)c3)=O)CCC2)nsc2ccccc12 C(CN=c1c(Br)c[nH]cc1[N+](=O)[O-])(C1CC1)NC(C1(COC)CCC1)=O c1(C(=O)NCC2C(NC(C3CN(S(N)(=O)=O)C3)=O)C2)cnnc2ccccc12 C=CCN=c1[nH]c(C(N2CCC(NC(C3CCC(=O)NC3)=O)C(O)C2)=O)cs1 C1(OCCCNC(C2CCC3CC23)=O)CCN(C(=O)C(F)=CC2CC2)CC1 CCCCC(C(=O)Nc1cnc(F)nc1)NC(=O)CCCC(OC)OC CC1(CNC(c2ccccc2CO)=O)CCN(C(=O)C(O)Cc2ccccn2)C1 n1(CC(=O)NCC(C)N(C(C(C)OCC)=O)C)c(C)cc(O)cc1=O c1(CNC(=O)C(F)CC2CCOC2)ccc(NC(C2CC23CCC3)=O)cn1 Cc1cc(OCCC(=O)NC2CC(C)(NC(C3CCC4(CC4)C3)=O)C2)cc(C)c1 N1(C(c2c(C)snc2)=O)CCC(NC(=O)COC(F)F)CC1C Cc1noc2ncc(C(N3CCC(NC(C4(C)CC4Br)=O)CC3C)=O)cc12 C1(C(=O)NCCOCCNC(c2nnn(C)c2C(F)F)=O)CN(CP(C)(C)=O)C1 CC(C(C)C(=O)N(CCCCCNC(c1cc2cccnn2n1)=O)C)C(C)(C)C c1(NCc2ccc(C(N3CCN(CC(C)C)CC3)=O)s2)cc(O)c(O)cc1O C=CCCC(C(=O)NCc1cccc(F)c1C)NC(=O)CC1CNC(=O)O1 C1(C(=O)NC(CCSC)C(=O)NCCCn2cnnc2)CC2CC(=O)C1C2 C1(C(=O)Nc2cc(C(=O)OC)c(Cl)cc2)CCCC(F)(F)CN1 N1(C(c2ncn(C)n2)C(=O)Nc2c(OC)cccc2)CC(OC)CCC1C N1(C(c2c[nH]c(=NC)o2)=O)CCCC(O)(CNC(=O)C(C)c2cccs2)CC1 CCC(O)C(=O)N1CC(O)(C(C)NC(=O)CNS(=O)(=O)C2CC2)C1 CC1CCCC(C(=O)NCCNC(C2CC3(CC3)C2)=O)C1 c1(C(N2C(CNC(C(CN(C)C)N(C)C)=O)COCC2)=O)cncc2c1CCC2 Cc1cc(C(N2CC(C)(C)CC2CNC(C2CCC(C)(F)CC2)=O)=O)cc(N)c1 c1(C(=O)NC2CN(C(c3cnc(C)[nH]3)=O)C(C)C2)cccc(Cl)c1O C#CCCCCCNC(=O)C(C1(O)CCC1)NC(=O)CCC=CC C12(C(=O)NCCN3CCN(C(C4CCCC4)=O)CC3)CC=CCN1CCC2 N1(Cc2c(OC)cc(Cl)cc2)Cc2[nH][nH]c(=NC(=O)c3nccs3)c2C1 N1(C(C(Cn2ccc(C)n2)C)=O)CC(NC(=O)Cc2cn(C)nc2C)C(C)C1 N1(C(C)=O)CC(CC(=O)NCc2c(C)coc2C)CC1(C)C.c1(C)cncn1C(C)C N1(C(c2ccc(N)cc2F)=O)CC2CC1CN(C(=O)CC1CC1(Cl)Cl)C2 C(=O)(C(C)CC(F)F)N1CCC(NC(C=CC(=O)N(C)C)=O)(CO)C1 C1(C(N2CC(NC(=O)CCn3cccn3)C(F)CC2)=O)CCn2ccnc2C1 c1(CCCN2CC(CNC(C3C(C)(C)C3)=O)OCCC2)cccc2nsnc12 C1(C2CCN(C(C3CCCCC3(C)C)=O)C2)(NC(c2cn(C)c(O)n2)=O)CC1 C=C(C)CC(C(=O)NC1CCC(N(C)C)C1)NC(c1cc(O)ncc1F)=O C12(CCCCC1)C(=O)N2.C1(C(N2CC3(C2)CC3(F)F)=O)(CO)CC12CCC2 C(=O)(C(CC(F)F)N(C(=O)CC1CC(=O)C1)C)NC(CCOC)C(C)C C1(CC(=O)NC2CC(NC(c3sccc3C3CC3)=O)C2)CCCC2(CCC2)O1 N1(CCCOC)CCC(C(=O)N(C)C(c2ccc(Cl)cc2)C2CCCN2)CC1 C#Cc1cc(F)c(C(=O)N(CC(C)(C)CNC(=O)CC(C)C)C)cc1F c1(C(=O)OC)cn(C)nc1NC(CNC(C1CCC(C)C1)=O)C(C)(C)C C1(NC(C2(C)CC(F)(F)C2)=O)CN(C(c2cocn2)=O)CCC1C(F)(F)F N1(C(CCc2c(C)noc2Cl)=O)CCN(Cc2csc(SC)n2)CC1C N1(C(c2cnn(C)c2F)=O)CCOCC(NC(=O)CCC2CCCC(=O)N2)C1 N1(C(C2C(C)(C)CO2)=O)CCOCC(F)(CNC(c2n[nH]cc2Cl)=O)C1 N1(CCNC(CNC(CC)=O)=O)CCC(NC(C2(C(F)F)CC2(C)C)=O)CC1 C1(C2(O)CN(C(c3ccc(C(C)C)cc3)=O)C2)(CNC(C=CC(CC)C)=O)CC1 CC1CN(C(=O)C(C)(C)n2cc(CO)nn2)CC1CN.S(=O)(=O)(C1CC1)NC1CC1 c1(C(=O)NCCC(C)(C)CNC(C2CC2(C)Br)=O)cccc2c1OCO2 CCCC(C)(C)C(=O)NC1CN(C(=O)COCc2cc(C)no2)CCC1F c1(C(=O)NC2(CNC(C=Cc3n(C)ccc3)=O)CC2)ncc(Br)cc1O N1(C(c2cccc(NCC)c2)=O)CCC(CCNC(=O)C(C)(C)CO)C(F)(F)C1 C1(NC(C(CCOC)C)=O)CCN(C(=O)Cc2sc(C)cc2C)CCC1(F)F c1(C(=O)NCCCC(C)NC(=O)C(C)(C)Nc2ccccc2)ncccc1Cl Cc1ccn2ncc(C(N3CC4CCC(NC(=O)CC5(C)CC5)CC4C3)=O)c2c1 C12(C(=O)NCCCCCN(C(C(CN(C)C)(C)C)=O)C)CCCCC1CCC2 c1(C(N2C(CC(=O)NC(C(=O)OCC)C3CC3)CC(F)C2)=O)nc(C)ccc1C N1(C(COC)=O)CCN(C(c2ccc(C)c(C)c2)=O)CCC1C.C1C(=O)N1C C1(CC(=O)N(CCCC(=O)NCC2C=CCCC2)C)CCC(=O)NC1 c1(CC)cscc1C(=O)N(CCCN(C(=O)C(C)OC(C)(C)C)C)C Cc1nc(C(=O)NCC2(c3ccccc3)CC(NC(C3CC3C#N)=O)C2)sc1C C1(CC(=O)NCC(CC)C(C)C)CCN(C(=O)C=CC(C)(C)SC)C1(C)C c1(CC)nc(C(=O)N(C)CC2CN(C(C3(C#N)CCCO3)=O)CCO2)c(C)o1 c1(C(N2C(CNC(=O)COC(F)(F)F)CCC2)=O)c(Br)ccc2c1OCO2 N1(C(C=CCCC)=O)CCN(C(=O)Cn2nc(C(F)F)cc2C)C2CC12 c1(C(CNC(=O)CCCC2CCC2)NC(C2(C#C)CCC2)=O)ccc(F)cc1F C1(NC(C(C)=C(C2CC2CC)C)=O)C=CC(CNC(=O)Cc2sccc2C)C1 c1(C(N2CCCC(CCNC(=O)CNc3ncccn3)C2)=O)cc(Cl)cc(Cl)c1 c1(OC)nccc(C)c1C(=O)NCCN(Cc1cccc(-n2cccn2)c1)CC c1(C(CC)=O)ccc(C(C)C(N2CC(NC(=O)C=CCOC)CC2C)=O)cc1 C1(CC(=O)N(C2CCN(C(c3ccc(Cl)cc3)=O)C2)CC)CCC(C(C)C)CC1 C(c1cnc[nH]1)=C(C)C(=O)N(CCCN(C)C)CCNC(C1(C(C)C)CC1)=O c1(CC)c(C(N2CCC(C)C2CNC(=O)CCc2nc(C)c(C)[nH]2)=O)ccn1C N1(C(CN(S(CC)(=O)=O)C)=O)CCCC(c2nc(C)n(C)n2)C1.C(C)(C)C C(=O)(C1=C(C)CCCC1(C)C)NCC(C1CCOC1)NC(C(C)NC(CC)=O)=O C(=O)(C(CNC(C1CC2(CCC2)CO1)=O)C(C)(C)C)N1CC(OC)(CO)C1 n1(CC(=O)NCC2CCCN(C(c3cn(C4CCC4)nn3)=O)C2)cnccc1=O C12(C(N3CCN(C(CN(C)C(c4csc(O)n4)=O)=O)CC3)=O)CCCC1C2(F)F C1(C(N2C(CN(C)C(c3ccc(C)cc3OC)=O)CCC2)=O)CCN(OC)CC1 C(=O)(C1=CCC2CCC1N2C(C12CCCCC1C2)=O)NC1CCN(C)CC1 CC(CN=C(NCCF)N1CCC(C(F)F)C1)N(C)C c1(C(=O)NCC23CC2CN(C(c2cc[n+]([O-])cc2)=O)C3)cnc(C(F)F)cn1 Cc1nc2n(n1)CC(C(=O)NCC1(O)CCN(C(C3(CCF)CC3)=O)CC1)CC2 C(C(C)C)(C(O)C(=O)N1CC2CC2C1C(=O)NC1CC(=O)N(C)C1)OC CC1CCc2[nH]c(C(=O)Nc3ccc(N4CCCCC4)cc3)cc2C1 N1(C(C(C)SCC)=O)CC(C)(C)C(NC(=O)C(C)SC)C(C)(C)C1 N(C(=NCC(CC1CCCCC1)CO)N1CCC(C)(C)CC1)CC(C)(C)C c1(C(=O)NC2C(CO)CCN(C(C3(C)CC(=C)C3)=O)C2)ccc2c(c1)CC(=O)N2 N1(C(c2c(OC)scc2)=O)CCCN(c2ccc(COC(C)C)cn2)CC1 c1(CC(N2CCC(COC(F)(F)C(F)F)CC2)=O)ccccc1C(F)(F)F C1(NC(c2c(C(C)C)n[nH]c2)=O)CCC(C)(CNC(=O)Cc2nnc(O)s2)C1 c1(C(=O)Nc2ccsc2C(=O)Nc2csc(C(F)(F)F)n2)ccc(O)nc1 C(CN=c1[nH]cc(Br)cc1C#N)C1CC(NC(C2(SCC)CC2)=O)C1 N1(C(=O)NC)CCCC(NC(=O)CCSSN)C1.c1(NC2CCCC2SC)nccc(OC)n1 CC1CN(C)CC(C(N2CCCC2CNC(c2ncccc2OC(F)F)=O)=O)O1 C1(CN(CC(=O)OC)CCNCCOCCO)CCC(=O)CC1 c1(C(=O)NCC2N(C(COCCCOC)=O)CCC2(C)C)ccc([N+](=O)[O-])n1C N1(C(c2c(C)coc2)=O)CCCC2(CCC(NC(C3(CO)CCCC3)=O)C2)C1 c1(-c2c(C)occ2)cc(=NC(=O)C(=O)OCC(C2CCC2)C2CCC2)[nH]o1 c1(C(C(=O)NCC(C)NC(c2cnco2)=O)(F)F)ccc(OC(C)C)cc1 C12(CC(=O)NCC3CC3CNC(c3ncncc3Cl)=O)CCC(CC1)OC2 C1(NC(C(C(CC)O)C)=O)CCC12CCN(C(=O)COC1CCCCCC1)CC2 C(C(=O)NCC1(F)CCN(C(C2CC(=C3CCC3)C2)=O)C1)(C(C)C)SCC Cc1ccc(C(=O)NCC2CN(C(=O)C(C(C)C)N(C)C)CC23CC3)cc1C C(=O)(C(F)C(C)CC(C)(C)C)NC1C(c2onc(CC)n2)CCCC1 C12(NC(c3coc(OC(F)F)n3)=O)CCCC1N(C(C1CCCCS1)=O)CCC2 C1(CNC(c2c(C)nc(C(C)C)o2)=O)CN(C)CCN1C(=O)C=CC(C)C c1(CSC)nc(N(CC(O)CN(C)C(c2coc(C(F)F)n2)=O)C)cc(Cl)n1 C1(NC(=O)CCc2cncnc2)CCC(O)CN(C(=O)CC2CCCCC2O)C1 Cn1ccnc1CNC(C1CCCC1)NC(c1nc(C(F)F)no1)C c1(C(N2CCC(NC(C(C)OCC=C)=O)(CF)C2)=O)cnc2onc(CC)c2c1 C(CC(C)(C)CNC(=O)COC1(C)CCC1)NC(c1c(C)cno1)=O c1(CNc2ccnc(C(=O)OC)n2)ccc(-c2ccc(CO)c(OC)n2)cc1F CCCC(CNC(c1ncncc1Cl)=O)C(=O)NC1CCOC1 CCC(CC(=O)N(CC(=O)NCCC(C)F)CCOC)C(C)C C(c1ccccc1C#N)=CC(N1CC(C)C(NC(=O)C=Cc2ccn(C)c2)C1)=O c1(CC)cc(C(=O)NCC2CC(NC(c3cc(C(F)F)n(C)n3)=O)C2)ccc1Cl C(=O)(CCCCCCNC(=O)C(C)N(C(=O)CC)CC)NCC1(CCC)CCC1 N1(CC)CC(CNC(=O)Nc2cn(C)nc2OC(C)C)CC1=O c1(C(CC)N(C2CCCC2)Cc2nnnn2C(C)C(=O)OC)cc(F)cc(Br)c1 C(=O)(C(F)CC(C)(C)NC(=O)CC1(C)CCC1)NC(c1cn(CC)nc1)C C1(C(N2CCN(C(=O)CN3CSCCSC3)CC2)=O)CCn2nccc2C1 CC(C)CS(=O)(=O)CC(=O)NCCCCC(C)NC(C1OCCN(C)C1=O)=O N1(C(CN(CCOC)C)=O)CCCC(O)C1.c1(C)occc1F.OC C(=O)(C(C)(C)C(=O)NC(c1cccc(Cl)c1)CNC(c1sccc1C)=O)OC Cc1cc(=NC(C)CC(C)O)[nH]c(NCCc2cc(O)n[nH]2)n1 c1(NC(=O)Cc2cnccn2)ccc(NC(c2ccoc2C2CC2)=O)cc1F C(C(C)(CC)C(N)=O)N(C(N1CCC(C(C(=O)OC)O)C1)=O)C(C)C c1(NC(C2N(C(C(C)CO)=O)CCC2)=O)ccc(I)nc1 C1(NC(CCCn2ncc(C)c2)=O)CCCCN(C(=O)CC2CCNC(=O)C2)C1 c1(CC)cc(Cl)ccc1C(=O)NCC1CC(C)(C)CN1C(c1cc(C)c(Cl)s1)=O c1(CN(C(=O)C(C)(C)OC(F)(F)F)C)ccc(C#N)c(F)c1 C(C(C)(C)CC(=O)N1CCCCC(NC(=O)C=Cc2ccncc2)C1)N(C)C N1(C(c2ccc(=N)[nH]c2)=O)CCC(NC(c2cc(F)n[nH]2)=O)C(F)C1 C1(CNC(CC(=C)C)=O)CC(O)CN1C(=O)Cc1ccc(OC)s1 c1(NCC(=O)NCCC2CCCN2C(=O)C(F)OC(F)(F)F)cccnc1 c1(OC)ccc(C=CC(=O)NCC(C)N(C(=O)CC2CCOC2)CC)cc1 C(=O)(C(C)C(C)COC)N1CCC(C2N(C(c3c(CC)scc3)=O)CCC2)CC1 C(=O)(C1CCCc2cccnc21)NCC1(NC(CCCC#N)=O)CC1 C1(C(=O)Nc2cncc(C)n2)CC2CCC1N(C(c1cc(I)ccc1Cl)=O)C2 C=CCC(CC(C)C)C(=O)NC1C2CC(NC(=O)CC(O)C3CCCC3)CC12 C(=O)(C1CS(=O)(=O)c2ccccc21)N1C2CN(C(=O)CCC3CC3)CC1CCC2 C1(NC(CC2COCC(C)(C)O2)=O)CCC2(CC1)CN(C(C1CCCOC1)=O)C2 c1(CCC(C)=O)cn(CCN(C(=O)CCn2ccnc2)C2CC2)nn1 CC(C)C(C(C)NC(C1(CCF)CC1)=O)NC(=O)COCc1cccc(Cl)c1 c1(C(=O)NC2CCN(C(=O)C3=CCCCCC3)C2)ccc2c(c1)C(=O)NCC2 C12(CCCCC1)C(=O)NC2.C(=O)(CCCOCCOC)NCC=C Cc1cccc2c(C(N3CCC4(CC3)CC4NC(=O)C(C)(Cl)Cl)=O)csc12 c1(C(=O)NC2C(CNC(CNC(=O)CC(F)(F)F)=O)CCC2)cc(F)cc(F)c1 C=CCC(C(=O)N1CCC(C(C)C(N2CC3(CCCN3C)C2)=O)CC1)C(C)C C(C(=O)N1CC2(CNC(C3C(OC(C)C)C3C)=O)CC1CO2)(C(C)(C)C)SC N1(C(CCn2nc(C)c(Br)c2)=O)CCC2C(C1)CN2C(=O)CCC(N)=O C(=O)(C(F)(F)C(C)O)N(C(C)C(=O)Nc1cn(CC2CC2)nn1)CC1COC(=O)C1 n1(C(C(=O)NCCC(CNC(COCCCC#C)=O)O)C)ccc(C2CC2)n1 N1(C(c2nnn(C)c2N)=O)CCCN(C(=O)CSc2nncs2)C(CO)C1 N1(C(c2cccnc2C2CCC2)=O)CCC2(CCN(C(=O)CC3CCC3)C2)C1 C1(NC(c2ccsn2)=O)CC2CC1CN(C(C1(C(F)F)CCCO1)=O)C2 c1(C(N2C(C(C)(C)C)CCC2)=O)coc2c1CN(C(=O)CC1CSCCO1)C2 C1(=O)C(C(C)(C)C)CN1.CN(S(N)(=O)=O)CC(=O)Nc1cn(CCC#N)nn1 N=c1nc(O)c(CC(=O)NC(CNC(=O)CCN2CCCS2(=O)=O)C2CC2)c[nH]1 C1(CNC(COC2(C)CCCC2)=O)CCN(C(=O)C=C2CC2)CCC1(F)F N(C(=NCCCNC(c1cccnc1)=O)NCC(C)(C)C)CC(C)C C=C(C)CC(C)C(=O)NCC1(NC(C2CN(C(=O)OC(C)(C)C)CC23CC3)=O)CC1 C(c1cccnc1C)=CC(=O)NCC1(OC)CCN(C(c2c(CC)[nH]cc2)=O)C1 Cc1nn(C)c2nc(C(=O)NCC3CC3NC(=O)CN3CCC(C)(O)C3)ccc12 C1(C(N2CC(CNC(C(=Cc3ccccn3)C)=O)C2)=O)CCS(=O)(=O)N1C Cc1ccc(C(N2CCCC(NC(C3CN(C)C(=O)N3)=O)C2)=O)cc1 c1(C(=O)NCC(CNC(c2ccc(OC)cc2Cl)=O)(C)O)n[nH]c2c1CCCC2 N1(C(c2c(C)cc(C(F)F)o2)=O)C2CCCC1CN(C(c1cnco1)=O)C2 c1(C(N2CC3C(NC(C(F)=C(C)C)=O)C3C2)=O)ccc2nnn(C)c(=O)c2c1 C(=O)(CC(F)(F)C(F)(F)F)N1CC(CC)(CC)OCC1 C(=O)(C(CC(C)(C)C)OC)NCC1CN(C(CCCN(C(=O)OC)C)=O)CC1O c1(CCC(=O)NCC2(NC(CCC(C)(C)F)=O)CCOC2)n[nH]c2ccccc12 c1(C(N(C2COC(C)C2)CC)=O)ccc(CNC(=O)C2CC2)nc1 c1(CCC(=O)N(CCCOCCNC(C2(O)COC2)=O)C)cccnc1Cl C(=O)(CCC(=O)NN(C)C)NC(C1CN(C(c2cc(C(C)=O)oc2)=O)C1)C CC(Cc1ccccn1)C(=O)N1C(CO)C(=O)C2(CNCOC(C)(C)C)CC1C2 N1(c2ncc(C(=O)OC)s2)CCCC2CN(C(=O)CCNC(C)=O)CCC12 c1(C(N2CCCN(C(C3(F)CCC3)=O)CC2CO)=O)cnc2ccccn12 C(CNC(=O)C(C)(F)F)(C(=O)NC(CC1CCCC1)CO)N(C)C C1(F)(CNC(=O)C=C(Cl)Cl)CCCN(C(c2cc(Cc3ccccc3)[nH]n2)=O)C1 c1(C(=O)NCC2C(NC(CN(C(C)=O)C)=O)CCC2)ccc(F)c(C(C)(C)F)c1 c1(CNC(=O)CCCc2ccc(F)cc2)ccc2c(n1)OCCO2 CN1CC(NC(C2(CCNC(C3(C)CC(F)C3)=O)CC2)=O)CCC1=O C1(NC(C=CC=CCC)=O)CCN(C(=O)CC2(CSC)CC2)C(C)C1 C1(F)(CNC(CCNC(N)=O)=O)CCC(NC(=O)CSc2ccncc2)C1 CC(O)(C(=O)NCCCOCCNC(c1cn(CC(N)=O)nn1)=O)C1CCC1 C(=O)(N=c1[nH]cc(C#N)cc1C)c1cc2cc(C)[nH]c2cc1 c1(C(C(=O)OC)O)cccc(Cl)n1.N1(CC2CCCO2)CCC(C)C1 c1(C(N(C2CCN(C(CCC#CC)=O)CC2)C)=O)cnc(OC)c(C)c1 Cc1cc(C)c(C(=O)NCCC(C)NC(=O)CCC2CCCC(=O)N2)c(N)c1 C1(C(=O)NC(C)C(=O)NCCCC(C)O)(OC)CC(C)C1 n12ncc(c1C)NC(=O)C13CC1CN(C3)C2=O.c1(C(=O)OC)ccc(OC)s1 C1(CC(=O)NC(CC2CCC2)C(=O)NCc2cn[nH]c2)CCCOCC1 C1(CCC(=O)OC)CCN(N2CCn3c(Br)cnc3C2)CC1 c1(CC)noc(CC)c1C(C)NC(C)CS(=O)(=O)C(=O)OC C#CC1CN(C(=O)C=Cc2ccn(C)c2)CCN1C(C1COCCC1C)=O C(C(C)(O)C(F)(F)F)NC(COC1CC(NC(c2nc(COC)oc2)=O)C1)=O C1(N(C(=O)COCC(F)F)C)CCC2CN(C(=O)CC3(C)CCC3)CC12 C(=O)(C(C)(C)C(C)(C)O)NC(C1(O)CN(C(CC(CC)c2ccccc2)=O)C1)C C1(C(N2C(CCC(=O)NCCC(=O)OCC)CCC2)=O)CCN(C)C1=O C12(C(=O)NC3CCCC3CNC(=O)C(F)(F)C(F)F)CCCCN1CCC2 CS(=O)(=O)C1CC(NC(C2CCCN(C(c3ccc(Cl)c(Cl)n3)=O)C2)=O)C1 N1(C(C)=O)CCC(NC(C2CCCN2C(C2CC(CC3CCCO3)C2)=O)=O)CC1 C1(N(C(c2cc(CNC(C(C3CCOCC3)C)=O)[nH]n2)=O)C)CCC(CO)CC1 NC1CS(=O)(=O)C2CN(C(c3c(C(F)F)cccc3F)=O)CC12 C1(OC)CC2(CCN(C(C34CC(C)(CN3C(=O)C#CC3CCC3)C4)=O)C2)C1 CC1=C(C(=O)NCC(C(=O)NCCc2cccs2)C(C)C)CCCO1 N1(C(C2CCN(CC)C2)=O)CCC(NC(C2CCCC(=O)N2CC)=O)C(F)C1 c1(C2CCN(C(c3c(OC)scc3)=O)C2)ccc(C)cc1 C1(C(=O)NCC2CCN2C(=O)C2=CCOC2)CCc2ncnn2C1 N(C1CCCn2ccnc21)C(C1C(C)(C)C(NC(=O)Cn2ccnn2)C1)=O c1(C(=O)NC(C(=O)NCCOCCC=C)CC2CC2)ncncc1N C1(CCNC(C2C(CCC)C2)=O)CCN(C(=O)C(C)CC2CCCO2)CC1(F)F N1(C(CC2CC(NCc3n(CCC)ccn3)C2)=O)C(CO)CCC12CCC2 N1(C(c2nc(COC)sc2)=O)CCC2CN(C(=O)C(n3ccnc3C)C)CC12 c1(SCC(=O)N(C2CCS(=O)(=O)C2)CCOC)ccc(N2CCCS2(=O)=O)cc1 c1(C(=O)NC2CCCC2NC(CC2C(CSC)C2)=O)ccc(-c2cscn2)cc1 c1(C(N2CC3(CN(C(C(C=C)O)=O)C3)C2)=O)cccc2ccc(Br)nc12 C(=O)(C1=NN2CCCN=C2N1)NCC(CNC(C(c1c(C)noc1C)C)=O)O C1(NC(c2c(C)cc(C)nc2)=O)C(C(C2CC2)NC(c2cscn2)=O)CCC12CCC2 c1(OCCC(=O)NCCCCNC(c2cccn(O)c2=O)=O)ccc(F)c(F)c1 C1(C(N(c2cc(CF)on2)C)=O)CCN(C(=O)CCC(=O)N2CCOCC2)CC1 C1(C(=O)NCc2c(C(=O)NOC3CCC3)cccn2)CCCC(=O)N1 C=C=CC(C)C(=O)NC1(CCNC(c2cnccc2C(C)(C)C)=O)CCC1 CN1CCCCC1CCC(N1CCC(C)(NC(=O)CC2CCC(C)(C)O2)C1)=O C#Cc1ccc(N(C(C(=O)NCC2CC2)C)C(=O)CSCC(F)F)cc1 N1(C(c2[nH]c3cc(C)oc3c2)=O)CCCC2(CCN(C(c3coc(O)n3)=O)C2)C1 n1(CCCSC)nnnc1C(C)(CC1CCCO1)NCC(Cl)(Cl)Cl CC1=C(F)CN(C(C2CN(C(=O)CC3(C)CCC3)CC2C(C)C)=O)CC1 C1(CNC(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC(C)F)CC1(F)F C1(C(=O)NC2(C)CCN(C(c3n(CC)ccn3)=O)C2)CCc2ncnc(C)c2C1 Cc1ccc(C2CC2)c(C(=O)N(C2CCCN(C(=O)CCC(N)=O)CC2)CC)c1 C1(NC(C(C)=CC2CC2)=O)C2CCC(C2)C1C(=O)Nc1cc(F)ccc1O Cc1csc(C(F)(F)C(=O)NC(C)CC(C)NC(c2cccnn2)=O)n1 Cc1c(Cl)ccnc1C(=O)NC1CC(NC(=O)CN2CC3CCC2C3)C1 Cn1cnc2[nH]c(C(N3CCC(NC(c4ccc(Br)o4)=O)C3(C)C)=O)cc12 N1(C(C(=O)NC(C)C)C2CC2CC)CC(C)(C)C1c1ccccc1 N1(C(c2c(SC)scc2)=O)CCC2CCC(C1)N2C(C1CCCOC1C)=O c1(OCC(=O)NCCCC(C)NC(=O)CCC2CCC2)cccc(N)c1 C=CCCCCC(=O)N1C(C(=O)NC(C2CCCCC2)CC)CCC1C(C)C N1(C(C2C(C(=O)OC)CC2)=O)CC2(CCCC2NC(=O)CCCC(C)=O)C1 C1(C(=O)NC2(C)CC(NC(CCCOCC)=O)C2)CCCC2(CN(C(C)=O)C2)O1 N1(C(C2C(C)C2)=O)CCCC(NC(c2c(Cl)nsc2Cl)=O)C1 c1(C(=O)NCCNC(C2CCC(C(F)F)NC2=O)=O)ccc2nnc(S)n2c1 Cc1cc(N2CCOCC2)nc(=NCC2CCCN2C(=O)CS(=O)(=O)C2CC2)[nH]1 N1(C(c2c(OC(CC)C)cccc2)=O)CCc2c(C(=O)OC)cc(Br)cc21 N1(C(c2cccc(OC)c2)=O)CC2CC(CNC(=O)C(N3CCOCC3)C)C2C1 N1(C(C)=O)CCOCC1C(=O)NCC12CC(C1)N(C(=O)C1=C(C)CC1)C2 C=CCCCCCCC(=O)NC1CC(CO)N(C(c2cnc(S)[nH]2)=O)C1 C(=O)(C(C(C)C)NC(c1ccoc1)=O)NCCC1CN(C(C2(C=C)CCC2)=O)C1 N1(C(C2(OC)CC(C)(C)C2)=O)CCCCC(C(=O)NCC(F)(F)CO)C1 N1(C(CCOCCOCC)=O)CC2CC(C1)N(C(c1ccoc1C(F)(F)F)=O)C2 c1(C(N2C(C(C)NC(C3CCCS3)=O)CCC2)=O)cn(C)c2ccc(Cl)cc12 C1(NC(=O)NC(c2nn(C)cc2O)C)CC(C)CN(C(=O)OC(C)(C)C)C1 c1(C(N2CC(C(C)NC(C(=O)NCC)=O)C2)=O)ccc(Cl)c2ccccc12 C1(C(=O)NC(CCC)C(N)=O)CC1C1CN(C(=O)CC2COCCOC2)C1 CN1CCN(C(=O)C(=O)NC2CC3CCC2NC3)CC1(C)C Cc1ccc(CC(N2CCN(C(=O)Cc3c(Cl)cnn3C)C3CC23)=O)c(F)c1 C(=O)(C(CCC)CC(C)C)N(CCC)CCNC(C1(CCC)CCC1)=O C12(C(N3CCC(C(C)C)C3)=O)CC(CN1C(=O)C(C)CC1CCCC1)C2 C(CO)(CC(C)C)NC(=O)CCCC1CC(NC(C(CC)NC(N)=O)=O)C1 c1(C(=O)NCCCN(CCOC)Cc2nc(CC)sc2)cccc(C(N)=O)c1.SCC C(=O)(C#CC1(C)COC1)NCC=CC(=O)N(C1CCCCC1)CC C(CCC(C)C)(C(=O)N1CCCC(OC2CC2)C1)NC(CCC(CC)OC)=O CCCCCC(C)CC(=O)NC(C)CCN(C(=O)Cc1coc(C(F)F)n1)C Cc1cn2nnc(C(=O)NC3CC3NC(=O)CCc3nncn3C)c2c(O)n1 C1(C(=O)NC(C)CCN(C(=O)COC(C)(C)C(F)(F)F)C)CCCCN(C)C1=O N1(C(=O)NCCC)CCC(C)(C(=O)NC2CCCC2C(N)=O)C1 c1(C(N(C)C)=O)ccccc1C(=O)NCC1CCCCC1NC(C1CC12CC2)=O N1(C(CCN(CC)CC)=O)CCC(C(F)F)(CNC(C23CC(C)C2C3)=O)C1 CCCC(C)(CNCC(F)(F)CCNC(=O)CCCCC(C)C)CCC N1(S(c2c(NCC3(SC)CC3)nccc2)(=O)=O)CCc2c(ccc(Br)c2F)C1 c1(OC)cc(C(N2CCC(C)C2CNC(=O)C2=CCOCC2)=O)ccc1Br C1(NC(Cc2c(C)noc2Cl)=O)CCN(C(C2CC(=O)N(C3CC3)C2)=O)CC1C N(C(=NCc1cc(C)on1)NCc1cn(C(C)(C)C)nn1)C(CC=C)C C1(NC(C2C(C)OCC2)=O)CC2CCC(C1)N2C(c1cccc(CO)n1)=O N1(C(=O)Nc2ccc(C(OC)OC)nc2)CCS(=O)(=O)CCC1C(C)(C)C Nc1cccc(C(=O)NC(CNC(=O)CCc2cscn2)CC(F)(F)F)c1O C(=O)(C(O)P(C)(C)=O)NCC1(C)CCCC1NC(=O)CCCCCl Cc1ccncc1CC(=O)NCc1cnn(C)c1C(=O)NCCc1cncs1 CCCC(C(=O)NC(C)Cc1cccc(Br)c1)OCC CN1CCc2nc(C(N3CCC(CCNC(=O)Cc4cnc[nH]4)C3)=O)sc2C1 N(C1CCCc2ncc(C(F)(F)F)cc21)C(COc1cc(OC)c(Cl)cc1)=O C1(C(=O)OCC)CN(C(=O)C(C)(C)CC)CCC12CN(C(=O)C(C)NC=O)C2 C1(C)(CC(=O)OC)CCN(N2CC(NC(c3cccc(F)c3C)=O)C2)CCO1 C1CCCCCC(=O)N1.Cc1ccc(CCc2cn(CC(=O)O)nn2)cc1 Cc1ccccc1CC(N1CCC1C(=O)NC(c1c(C)n[nH]c1C)C)=O c1(OC)ccc(-c2nc(CC=Cc3ccccc3)nn2CCC(C)(C)OC)nc1 N1(C(C(C(C)C)=O)=O)CC(C2CCCCN(C(=O)CC3CSC3)C2)C1 N1(C(c2cc(CCC)[nH]n2)=O)CC(C(=O)NC2CCC(=O)NC2=O)C(F)(F)C1 N1(C(C(C)n2cccn2)=O)CCCN(C(c2cc[nH]c(=N)c2Br)=O)C(C)C1 C(=O)(C(CCN(C)C)NC(c1ccsc1C)=O)NCc1c(COC)noc1 c1(C(N2CCCC2c2cn(C3CC3)nn2)=O)ccc(O)c(CO)c1 c1(C(N2CC(C)(NC(c3cc(CF)on3)=O)C2)=O)cnn2c(N)ccnc12 c1(C(=O)NC2CCCC(NC(C3(CCC)CC3)=O)CC2)cc2ncccn2n1 C12(C(N3CC(NC(c4n(C(CC)C)ncc4)=O)C(OC)C3)=O)CC1COC2(C)C c1(CC(C)C(=O)NCC2CCCCN(C(=O)C(F)(F)C(F)F)C2)ccc(Cl)cc1Cl CC(CC(C)(C)C)C(=O)N1CC2C=CC1C(C(=O)NCC(F)Br)C2 N1(C(C2N(C(CSCC)=O)CCCC2)=O)CC2CC(C)C2C1 C123COCC1CN(C2)C3=O.C12CC(OC)CN1C2=O.C(=O)(CC(=O)OC)NCC Cc1cc(C)c(C(=O)NC(CNC(c2c[nH]cc(Cl)c2=O)=O)C2CC2)cc1Br C=CCCN=C(NCCCSc1ccccc1[N+](=O)[O-])NCC1CCOCC1OC c1(SC)cccnc1C(=O)NC(c1ccnn1C)CNC(=O)C(C)CC1CCC1 c1(NCC(CCNC(=O)C(=O)NC2CCNC2)OC)c(C(F)(F)F)cnn1C C1(C(C)C)CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CC2CCCC(=O)N2)CC1 C1(CNC(C2C(CCC)C2)=O)CC(NC(c2cccs2)=O)CO1 N1(C(c2c(COC)noc2)=O)CCN(C(c2ncn(C(C)(C)C)n2)=O)CC1 Cc1ccc(-n2nc(Cn3cccn3)nc2CC2(C)CC2(F)Cl)cc1C C1(C(=O)NCC2CCN(CC)CC2)CCC(C)N(C(=O)Cc2cncnc2)C1 CC(C)C(O)C(=O)NC1CC(F)(CNC(c2ccc(CC(N)=O)cc2)=O)C1 c1(C(N2CCC3CCN(C(C(CC)=CC)=O)C3C2)=O)ccc(C#CC2CC2)cc1 C(=O)(C(CN1CCOCC1)NC(=O)COC1CC1(F)F)OC(C)=CCCC1CC1 CC1(C)Cc2[nH]c3cc(Br)ccc3c2C1C(N1CC(c2ccon2)C1)=O C(=O)(C(C(C)C)C(C)C)N1CCC(OC)(CNC(C2C3CCCC23)=O)CC1 N1(C(c2ccccc2)=O)CCCN(C(c2ccc(CSC(F)F)o2)=O)CC1 C1(NC(c2nc(COCC)sc2)=O)CN(C(c2c[nH]nc2C)=O)CC(C)(C)C1 C1(NC(=O)C(c2cccc(Br)c2)O)C2CCC1CN(c1ncnc3occc13)C2 Cc1c(N)cc(C(N2CC(NC(c3cc(O)nc(Cl)c3)=O)CCC2C)=O)cc1N C1(C(N(C2CCC(NC(=O)CC(F)(F)F)CC2)C)=O)CC2OC1C1CC21 Cc1cc(NC(N2CCN(C(c3cc(C)n(C)n3)=O)CC2C)=O)cc(C)c1 N1(C(C2CCC(C)(C)O2)=O)CC2CC1CCN2C(c1nc2ccccc2[nH]1)=O n1(CCC)ncc(CNC(=O)C(c2ccc(C)cc2)C)c1Cl C1(C(=O)NC2(C)CCC2)CCCCCCN1C(c1occ2c1CCC2)=O CN1CCOCC1C(=O)NCCCN(C(=O)CCc1ccccc1F)CCO c1(C(=O)OC)c[nH]c(=NCC(C)CNC(C2(C)CC2(F)Cl)=O)cc1C CC(C(=O)N(OC(C)(C)C(=O)Nc1ccccc1)OC)n1cccn1 c1(C(=O)NC2CN(C(c3c(CCC)nns3)=O)C2)c(F)ccc(C)c1O C(C(C)C(=O)N(OC)C(C)C)NC(C(C)OCC)=O CCCCC(CNC(C1N(CC)CC1)=O)NC(=O)CCC(=O)N1CCC(O)CC1 C1(C(=O)NCCCCC(C)NC(Cc2c(C)scc2)=O)CN=C2N=CNN2C1 n1(CCC)nnnc1C(C(C)(C)NC(C)=O)NC(c1cnn(C)c1)C N1(C(C2C(CCOC)C2)=O)CC2CC(C)N(C(=O)CCc3ccccc3)C2C1 C(C(CC(C)C)C(=O)N1C2CCC1CN(C(=O)C(C)=C1CCCC1)C2)OC N(C1CCC(NC(=O)C(=O)C(C)(C)C)c2ccccc21)C(c1scc(C)c1)=O N1(C(=O)CCn2cccn2)CCOC2(CCN(C(C3(O)CC3)=O)C2)C1 c1(CNC(=O)NC2CCCC2n2cc(Br)cn2)cccc2ccoc12 C12(NC(C3CC(=O)N3)=O)CCC(C1)N(C(c1ocnc1C1CC1)=O)C2 C1(C(F)(F)F)(NC(=O)NCc2c(CC)non2)CCN(C)C1 n1(CCN(C(=O)Cc2cc(C(F)(F)F)ns2)CC)cc(-c2csnn2)nn1 Cn1nnc2c(C(=O)NC3CN(C(=O)CP(C)(C)=O)C4(CCCC4)C3)ccnc12 CN1CCCCC(C(N2CC(NC(C3(C(C)(F)F)CC3)=O)CC23CCC3)=O)C1=O CS(=O)(=O)CCC(=O)NC1CC2CC1N(C(=O)Cc1ccsn1)C2 c1(C(=O)NCC(CNC(CC(=C)Br)=O)(C)C)cc(C)c(C)c(S(N)(=O)=O)c1 C(CCCCCC(=O)N1CC(C2CN(C(=O)COCCF)C2)C1)SC N1(C(c2cnc(SC)s2)=O)CC2OCCN(C(c3cnc4occc4c3)=O)C2C1 C(=O)(CC1CCOc2ccccc21)N1CC(NC(C(C)SC)=O)C(C)C1 C1(C(C)C)CCC(C(=O)Nc2cnc(C3CC3)nc2)N1C(=O)CCCn1cccc1 c1(CNC(C(C=C)C)=O)cccc(CNC(=O)C=CC)c1.C1(S)CC(F)(CSCC)C1 C=C(C)CCC(=O)N1CCC(O)(CNC(C2CCN(c3ccncc3)C2)=O)C1 C1(CC(=O)NC(CNC(Cc2c(C)nsc2)=O)C)CCCCCC1 c1(OC)ccc(C(=O)NCC2CC2CNC(=O)C(CNC(C)=O)CO)cc1Cl c1(C(N(C2CCN(C(C(C)(C)F)=O)CC2)CC(N)=O)=O)cn2cccnc2n1 c1(C(=O)NC2(C)CCN(C(=O)Cc3csc(S)n3)C2)cccc2c1OCCO2 C1(C(=O)NC2CC(COC)C2)CCN(C(C2CCCC2F)=O)CCO1 N1(C(C=CCCCCC)=O)CC(C(=O)NC2CCSC2)C(C(C)C)C1 C1(C)(CNC(CCCNC(CC2(C)CCC2)=O)=O)CCCCO1 CC(C)C(CNC(=O)C(C)N1CCCC1)NC(=O)CCn1ccnc1 CCC1=NOC(C(=O)N(CCCNC(=O)CC2CCCCCO2)CC)C1 Cc1c(C(N2CCOCC(C(=O)NCC(C)N(C)C)C2)=O)cccc1O N1(C(C2CN(C(C)=O)C2)=O)CCC(NC(=O)C(C)(C)C2CC2)C1Cc1ccccc1 Cc1ccc(Br)c(C(N2CCCC2CNC(C23CCN(CC2)C3)=O)=O)c1 S(=O)(=O)(c1c[nH]ccc1=NC1CCCOC1)NCC(C1CCOCC1)(C)OC CP(C)(=O)C1CCCCC1C(N1CCCC1(C)Cc1ccccc1)=O c1(OC)ccc(CC(=O)N(CCCNC(=O)CC2CN(C)C2)C)c(Cl)c1 C=CC1(C(=O)NCc2cnn[nH]2)CCN(C(C2CC(C3CC3)C2)=O)CC1 N1(C(C2(C=C)CCC2)=O)CC(C)CN(C(=O)C=CBr)CC1C c1(NC(=O)O)cnc(CNC2CC2c2ccc(OC)cc2)c(Br)c1.C1(CCN)(CC)CCC1 C1(O)(CNC(C23C(C(=O)OC)(CCC2)C3)=O)CCCN(C(c2cc(Cl)c[nH]2)=O)C1 CC1=CCC(NCCC(N2CCOCC2C2CCCCC2O)=O)CC1 N1(C(CCC2OCC(C)(C)C2)=O)CCC(O)(CNC(c2occc2Br)=O)CC1 C(CC(C(=O)NC(CO)C1CCC1)NC(c1ccn(C)c1C)=O)SC c1(C(=O)NC2CC(C)CN(C(C3(C)CCC34CCC4)=O)C2)ccn2c1CCCC2 c1(C(c2n(C(CC)C)nnn2)NCCCF)ccc2c(c1)C(=O)NC2=O CCC(C)C(C(=O)N1CC(NC(=O)CCc2nnc(C(C)(C)C)o2)C1)NC(C)=O c1(CC)nc(C)c(Cn2cc(C3CCCN3C(C3CN(C(C)=O)C3)=O)nn2)o1 Cc1cccn2c(C(N3CCC4(COC(CNC(=O)C(C)O)C4)C3)=O)cnc12 c1(C(C(=O)NCC(C)CNC(=O)C(O)C2CCC2)F)ccccc1F C=CCC(C)(C)CC(=O)NC(C)C(N1CC(C2CC2)(OC)C1)=O Cc1ccc(Br)c(C(=O)N(C2CC(NC(C3CC4(CCC4)CO3)=O)C2)C)c1 C1(CNC(CCc2n(CC)ccn2)=O)C2CN(C(=O)CCCCC3CC3)CC12 C1(O)(CN(C)C(C2CCC(F)(F)C2)=O)CCN(C(=O)CCc2cc(Cl)no2)C1 C1(Oc2cc(C(=O)OCC)[nH]n2)CCC(F)(F)CC1.C1(N)C2CN(C(=O)CO)CC12 c1(CCC)ccc(N)c(C(=O)NCC2CCCC2NC(=O)CC2CC=CC2)c1 c1(CC(C)C)nc(C2CC2)nn1CC(F)(F)F.c1(C2C(C)C2)cccc(Cl)c1 C1(NC(CC2CC(C)(C)C2)=O)CC2CC1N(C(=O)CCc1nc(C3CC3)no1)C2 CC(C)CC1C(=O)N(C)NC(=O)N1.c1(Cc2nc(CN)no2)ccccc1 Cc1nnc(C(C)NC(=O)C(Cn2cncn2)NC(=O)CCCNC(N)=O)s1 c1(C(=O)NCC2OCC(CNC(c3ncn(CC)c3)=O)C2)c(C)ncn1OC C(C)(CCC(=O)NC1CC(=O)N(C2CN(C(=O)COC)C2)C1)OCC CCS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CCC2NC(C2CC2C(C)C)=O)c1 C1(COC)CN(C(=O)Nc2cnc3n2CCOC3)CC(C)(C)O1 N1(C(C2CCC(=C)CC2)=O)CC(OC)CC1(C)CNC(C1CN(C(C)C)C1)=O c1(C(C(=O)Nc2ccccc2Cl)NC2(C)CCCC2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC2(OC)CN(C(c3cccn(C)c3=O)=O)C2)nnc(O)cc1O C(=O)(C(CC)CC(C)C)NC(C1(O)CCN(C(Cc2c(C#C)cccc2)=O)C1)C C(N=c1[nH]c2c(c(=NCCOc3cnccc3CO)[nH]1)CSC2)c1scc(CC)n1 c1(CCC(=O)OC)nc(Cl)cc(=NC2CCCN(c3ccccc3)C2)[nH]1 Cc1c(C(=O)NC(C)CNC(C2CC3C(C2)C3(F)F)=O)cc(C)c2ncccc12 N1(C(C2(c3ccn(C)n3)CC2)=O)CCOC(C(N2CC3CC2CS3)=O)C1 c1(C(N(CCCCN(C(COC(CC)C)=O)C)C)=O)ccccc1OC n1(CCC)cc(CNC(=O)C(CN(C)C)NC(c2nsnc2O)=O)cn1 N1(C(c2scc(OC)c2)=O)CC(NC(=O)CC2OCCC2(C)C)CC1C C1(C(=O)NCc2cn(CC)nc2)CCC2CCC1N2C(=O)CCn1ccnc1C c1(CC(=O)N(CC(C)(C)CNC(=O)Cc2c[nH]nc2C)CC)cnn(C)c1C CCCCCCC(CNC(C1CC1c1ccc(C)o1)C)CC CCCC(CCCNC(=O)CCc1cnn[nH]1)NC(c1scnc1C(C)C)=O N12CCCC(C(F)C1)NC(=O)C=CC2=O.C(=O)(CC(C)(C)C)Nc1nc(C)sc1 N1(C(c2c(C)cccc2)=O)CCC2(C(N3CC(n4ccnn4)C3)=O)CCCC12 N1(C(C=CCOC)=O)CC2C3CCC(C2C1)N(c1cc(-n2ccnc2)ncn1)C3 c1(C(N2CCC(CNC(C3(C)C(C)CCC3)=O)CC2)=O)ccc2oncc2c1 N1(C(C(CC)N(C)C)=O)CCC2(CCCN2C(c2cc(S(N)(=O)=O)ccn2)=O)C1 Cc1cn(C)nc1C(N1CC(CCNC(c2cc(C(C)(C)C)on2)=O)C1)=O C12C3CCC(C3)N1C(=O)C(=O)NC(=N)N2.C1(CCOC)CCCC(C)C1 C(C(CC(=O)N(C1CCCC(O)C1)C)NC(c1nc(C)c(C)s1)=O)OC N1(CC2CCC(C)O2)CCC=C(C(=O)N2CCOC(CCC(=O)N(C)C)C2)C1 N1(C(c2cccc(CSCC)c2)=O)CCCCC(NC(=O)CC2CC2(C)C)C1 CCC(C)C(=O)C(=O)N(CCCCC(=O)NCCn1ccccc1=O)C C(CCCC(CO)NC(C1CC2CCC(C1)O2)=O)NC(CC(C)F)=O c1(OCC)cc2ncnc(Nc3cccc(OCC)c3)c2cc1Br N1(C(C(CCNC(c2cccc(C)c2N)=O)O)=O)CC2(C1)CC(C)(O)C2 C1(NC(C2CC2c2ccncc2)=O)CC2CC1CN(C(c1c[nH]ccc1=O)=O)C2 c1(OCC(=O)NC(c2c(C)cccc2)C(C)(C)C)ccc(S(N)(=O)=O)cc1 C1(NC(=O)CC2CCCC23CC3)CCN(C(=O)C(O)Cc2ccccc2)CC1F N1(C(C23CN(C(c4c(OC)cccc4)=O)C(C2)CO3)=O)CC2CCOC(=O)C2C1 C1(C(=O)NCC2CN(C(C)=O)C2)CC2(CCN(C(c3cscc3C)=O)CC2)CO1 CCC(C)C(C)C(=O)N1CCC(O)(CNC(c2ccc(C3CCC3)nc2)=O)CC1 CC(C)C(CC(=O)NN=c1cncc(F)[nH]1)c1nccn1C N1(C(c2c(C)cc(C)o2)=O)CCCN(C(C2CC23CC3)=O)C(c2ccccc2)C1 C(=O)(C1CCCc2scnc21)NC(CCNC(c1c[nH]cc(C)c1=O)=O)C C(=O)(N=c1c(Cl)c[nH]cc1Br)C1C2(CCN(C(CCc3cn(C)nc3)=O)CC2)C1 c1(C(C)NC2COC(C3CC3)C2)cccc([N+](=O)[O-])c1 CC(C)CC(C)CC(C)C(=O)NC1CC(CNC(c2cncc(C(N)=O)c2)=O)C1 C1(C)(CC)CCN(C(=O)CCCCN(C(=O)CCCCC2CC2)C)C1 C1(CN(C(Cc2cc(OC)no2)=O)C)CCCC(NC(c2ccnnc2O)=O)C1 C1(C)(c2cn(C(C)C(=O)O)nn2)CCCN1C(c1coc(Cl)c1)=O N1(C(C=C(C)c2cccs2)=O)CCCCCC1CNC(=O)CC12COC(C)(C1)C2 c1(OC)csc(C(N2CC(CCNC(c3cn(C)c(C)n3)=O)C2)=O)c1OC N1(C(CC(CC)C(F)F)=O)CCC2(CC1)CN(C(=O)CC1CNC(=O)C1)CCO2 c1(C(=O)NC(CNC(C2(C=C)CCCC2)=O)C2CC2)sc2ccccc2c1C C(=O)(C(O)CCC(C)C)NC(CCSC)C(=O)NCc1ccc(Cl)nc1C c1(C(=O)NC2C(NC(c3nc(OC)oc3)=O)CCC2)ccc2c(c1)OC(C)(C)O2 C12(OC(C)C)CCC(N3CCN(Cc4ccc(Cl)cc4F)CC3)(CC1)C2 c1(C(=O)NC2CCN(C(c3[nH]c(=NCC)sc3)=O)C2C)cc2nc(Cl)ccc2o1 C(CCCN(C)C(C1CC(N(C)C)C1)=O)N(C(C=C(COC)C)=O)C C(CN=c1[nH]c(=NCCCOCC2CCOC2)c2sccc2[nH]1)=CCOC c1(C(=O)NC(CC(C)C)(C)CNC(=O)CC2OCCO2)cc2ccccc2s1 c1(C(=O)NC2C(C)C2C)c[nH]nc1CNC(=O)C=Cc1ccsc1 c1(SCC(N2CC(=C(CNC(=O)CCF)F)C2)=O)cccc(OC(F)F)c1 N1(C(c2cnc(CCCC)s2)=O)CCCC(C)(CNC(c2ccc(O)nn2)=O)C1 N1(C(C(C(C)OC)O)=O)CC2CCC1CN2C(c1sc(C)cc1C)=O Cc1ncc(C)c(=NCC2CN(C(c3ncc(Cl)cc3Cl)=O)CC2C(F)(F)F)[nH]1 C1(NC(c2c(OC)ccc(C(N)=O)c2)=O)CCCC12CN(C(C1CC1C#N)=O)C2 c1(OC)cccc(CC(=O)NCC(C)NC(C2CC3CC3C2)=O)c1 C12(NC(c3nc(CC)oc3)=O)CCC(CC1NC(C1(N(C)C)CC1)=O)C2 CC1CCCC1(C(=O)NCCCC1C=NNC1=O)NC(=O)Cn1ncn(C)c1=O N12CCc3sc(nc3C1)CNC(CC(C)C)C2=O.C(=O)(CCC(F)F)NC(C)C C=CC1CN(C(=O)Cc2cccc(Cl)c2Cl)CC1NC(c1ccccc1)=O C(=O)(C1=CC2(CCOC2)C1)N(CCCCCNC(c1n[nH]c(C)c1Cl)=O)C N1(C(CC2C(C)CCC2)=O)CC(NC(=O)COC2CCOC2)CC2(CCC2)C1 c1(CN(C(C2C(C)C2)=O)C)cnn2c1CN(C(c1cnc(C3CC3)s1)=O)CC2 N1(C(=O)NC(c2cc(Cl)sc2Cl)CC)CCn2c(CCO)nnc2C1 C(C)(C(C(C)C)NC(=O)CC1CN(C)C1)NC(c1cc(C)sc1)=O C(CCCCC(=O)NCc1ccncc1N(C)C)N(C(c1cc(C)oc1)=O)C C1(C(=O)NCC(CC(C)C)NC(=O)CCN2CCC(F)C2)CC2CC1C1CC21 c1(C(=O)NCC=CCNC(c2ccc(C(F)F)s2)=O)cc(C2CC2)ccc1F c1(CC)cc(C)c(C(N2CCCCC2CCC(C)(C)NC(=O)CSC)=O)o1 c1(C(N2CC(NC(CCCC(C)C)=O)C(C)C2)=O)cc2cc(Br)ccc2o1 c1(C(N(C2CCN(C(C3CCC(=O)O3)=O)C2)CCC)=O)cccc(C(C)C)c1 C12(C(N3CCCC(NC(C4(O)CCCCC4)=O)CC3)=O)C3CCC(CC13)C2(F)F Cc1cc(C(N2CCC(CC(=O)NC(C)(CO)C3CCC3)C2)=O)cc(O)c1 n1(CC(=O)NCC2CC(C)N(c3cc(Cl)ncn3)C2)ccc(O)nc1=O c1(C(N2CCC(c3nnc(C)o3)C2CC)C(=O)NC)ccc(Cl)cn1 C1(C(=O)NC(CC)(C)COC)CN(C(C2CCC2C#N)=O)CC12CCC2 Cc1cccn2c(=O)cc(SCC(=O)NCCc3cc4cccc(F)c4o3)nc12 C1(C(CNC(c2ccn(CC)n2)=O)(C)O)CCCN(C(=O)CP(C)(C)=O)C1 C1(C(N2CC(C#C)(F)C2)=O)CCN(C(=O)C(C#N)(CC)CC)C(C)(C)C1 c1(C2N(CC3N(C(=O)Cc4cc(C(F)(F)F)no4)CCC3)CC2)cccc(F)c1 C1(CNC(Cn2cnc(=N)[nH]2)=O)(CNC(c2ccccc2)=O)CCCCC1 c1(C(=O)NCC(C)(C)NC(C2CCc3ccnn3C2)=O)ccc2c(c1)COCO2 C=C(C)C(O)CC(=O)NCCC1(NC(c2cccc(SC(F)(F)F)n2)=O)CCC1 N1(C(C2(C=C)CCC2)=O)CCC2C(CCN2C(=O)Cc2csc(COCC)n2)C1 c1(C(N2C(CNC(CC3N(CC)CCC3)=O)CC2)=O)cc(=O)c2ccncc2o1 CC1CC(C(=O)NC2CCCCCC2C)CCN1C(C1CCCCC(=O)N1)=O N(C1CCCc2c1cnn2C)C(c1nnnn1CCCF)(COCC)C c1(CC(=O)N(C2(C(N3CCOCC3C(N)=O)=O)C(C)(C)C2)C2CC2)cccc(Cl)n1 c1(C(N2CCN(C(Cc3c(C)noc3Cl)=O)CC2C)=O)nccc2ccncc12 C1(NC(Cn2cc(C(C)=O)nn2)=O)CCC(NC(=O)CCC2CCCCO2)CC1 C1(CC(=O)NCCCCCN(C(C2(C(=O)NC)CCC2)=O)C)C(C)(C)C1(C)C c1(C(C)C)ccc(C(=O)NC2CC(O)(CNC(C3CC3c3cccs3)=O)C2)cc1 C1(CC=C)(NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CCN(C(=O)CN(C)C)C1 c1(C(=O)NCCC2(C)CCN(C(C3CC(N(C)C)C3)=O)C2)cc(F)cc(F)c1N N12CCCC(C)(C1)C2.c1(C(N(C(C)COC)CC=C)=O)ncc(CC)cn1 Cc1cnc(C(=O)N(C(c2ccccc2)CNC(C2(CC(C)C)CC2)=O)C)cn1 N1(C(c2scc(OC)c2)=O)CCOC(CCCNC(C2(CO)CC2)=O)C1 n1(CC)cc(Cl)c(C(N2CC3(NC(C4OCCOC4C)=O)CC2C3)=O)n1 c1(C(=O)NCCN(C(c2c(C)occ2C(F)(F)F)=O)C)ccc(F)c(C(F)F)n1 CC(O)(Cc1ccccc1)C(=O)N1CCC(Cc2c[nH]nc2OCC(F)F)C1 CN1CCC(CCC(=O)N(CCNC(c2ccc(C3CCC3)s2)=O)C2CC2)CC1 CCCC(C)(O)C(=O)NCC(C)N(C(=O)CCCN1CCCCC1)C CCCC(C)(C)C(=O)NC1C(OCCOC=C)CN(C(=O)C=CCOC)C1 CC1(C)CCCC(C(=O)NCCNC(=O)Cn2ncccc2=O)C1 N1(C(c2c(C)nc(-c3cccs3)o2)=O)C2CCCC1CN(C(=O)CCC1CC1)C2 C1(CC(=O)NC2CC(NC(C3(C)C(C(C)=O)C3)=O)C2)CC2CCC1CC2 C1(C(=O)NCC2CCOC2=O)(NC(C2C(C)CC2)=O)CC1(C)C C(CNC(c1cnnn1C)=O)(C(C)(C)C)NC(CC1(CSC)CC1)=O N1(C(c2cc(C(C)C)no2)=O)CC(C)(C)CC1CNC(c1cc(F)cnc1O)=O C(=O)(CCN=C(NCC(C1CCOCC1)F)NCC(F)F)N(C)C C(=O)(CCCCC(=O)NCCC(C)NC(=O)CCc1ccc2ocnc2c1)NC C(=O)(C(CC(=C)Cl)NC(=O)CCCCC#N)NC1(C)CC(=C)C1 C(=O)(CCCCC(=O)N1CCN(C(=O)C(C)NC(=O)NC)CC1COC)NC N1(C(C2(C#N)CC(C)C2)=O)CC2C=CC1CC2 CC(C)(C)CCC(C)(c1nnnn1Cc1ccccc1)NC1CC(C2CCC2)C1 c1(C(=O)NC(C2CCN(C(c3cccs3)=O)C2)C)ccc(C(C)(C)C)nc1 c1(C(=O)NCC2CCC(C(=O)NC(C)C(O)C(F)F)CC2)cc2ncccc2[nH]1 N1(C(c2cn3cc(C)sc3n2)=O)CCC(NC(C2COC(=O)N2)=O)C2(CCC2)C1 CC(C)CC(C(=O)N(C1CCC1O)C)N(C(=O)C1=CCSC1)C C(=O)(C(C(C)(C)C)C1CCC1)NCCN(C)C(c1ccc(C(O)CF)cc1)=O C(=O)(C(C)(CNC(=O)CCNC(c1ccco1)=O)CC)NCCOCC#C S(=O)(=O)(c1c[nH]ccc1=NCc1cncn1C)NCC1CCN(C(=O)NC)CC1 N1(C(C(C(C)C)F)=O)CCC(C)(C)C1C(=O)N(CC(C)(C)CN(C)C)C C1(C(=O)N(C)C)CC2(CCC2)CO1.CC(C)CC1CNC(=O)C2(CC2)C(=O)N1 C(CN=c1[nH]c(Cl)nc2ccccc12)C1CCCN(C(Cc2cc(C)no2)=O)C1 C1(=O)C(N(C)C)CCC(=O)C(=C)CCC(=O)NC(CC(C)C)CN1.OC n1(C(COC)C)nc(-c2ccc(C)o2)nc1C1COCCO1 C(=O)(C(C)CC(C)(C)C)N(CCC1CCN(C(CCCCC#C)=O)CC1)C C(=O)(C1OCCc2ccccc21)NCCN(C(CSC(C)C)=O)C1CC1 C(CS(=O)(=O)CC1CC1)NC(c1c(Cl)n[nH]c1C)c1n(CCOC)nnn1 c1(CC(=O)N(C)CC2CN(C(c3cn[nH]c3)=O)C2)sc(O)nc1O CC1(C)C(NC(c2cc(C#N)c[nH]2)=O)CCN1C(=O)CNS(N)(=O)=O N1(C(COC(CC)C)=O)CCCC12CCN(C(c1coc3c1CSC3)=O)C2 CN1CC(N(C)C(C23CC(NC(=O)CC(N)=O)(C2)C3)=O)CC1=O c1(C(=O)NCCN(C(CC(C)N(C)C)=O)CC(C)O)ccc2ccncc2n1 c1(C(C(=O)OC(CCOC(C2CC(O)CN2C)=O)=O)N(C)C)ccccc1[N+](=O)[O-] CC(CCN=C(NCC(F)F)NC1CCC(c2ccccc2)CC1)N(C)C.N1CCCC1 c1(OCC)ccc(C)cc1NC(C1C(CNc2ccc(COC)c(F)n2)C1C)=O C1(NC(c2c(C)c[nH]n2)=O)CCC(N(C(=O)CC(C2CC2)C2CC2)C)CC1 C1(C(=O)NCC(CC)NC(c2nonc2N)=O)CCC(O)C1 Cc1ccc(C2(C(=O)NCC(C)CNC(C3CCC(C(N)=O)O3)=O)CCC2)cc1 C(=O)(C(C)(C)CC(C)(C)C)NCC(C1CCN(C(C(C)C2CCC2)=O)CC1)(C)O c1(C(=O)NC(CCN(C(c2n(CC=C)ccc2)=O)C)C)nc(OC)ccc1Cl c1(NC(C2C(NC(c3cc(OC)nc(Cl)c3)=O)CCC2)=O)cc(Cl)c(Cl)cc1Br c1(C(C(=O)NC2COC2)NCOC(N(C)C)=O)ccccc1Cl.c12cn(nn1)CC2 c1(C(=O)NC(C2C(C(=O)NC3(C)C(C)C3)C2)C)cc(CO)n(C)n1 N1(C(CNC(=O)OC)=O)C2CCC1CC(OC(=O)NCCCO)C2 Cc1c(CNC(C2C3CC2N(C(c2ccc(NC4CC4)nc2)=O)C3)=O)nnn1C S(=O)(=O)(c1c(C)cccc1Cl)N(c1nc(C)c(F)cn1)C1CC(N)C1 N1(C(C2(C)CS(=O)(=O)C2)=O)CCC(O)(CCNC(c2ccc(N)cc2F)=O)CC1 c1(CCC(N2CC(C)CC(C(=O)OCC)C2)=O)ccc2c(c1)CCCN2C(C)=O C12(NC(c3c(C)n(C(C)C)nn3)=O)CN(C(=O)C=CC(C)C)CC1CS(=O)(=O)C2 N1(C(CC2C=CC(NC(CCNC(COC)=O)=O)C2)=O)CCCC1C#N CC1CCC(C(N)=O)CN1C(=O)CC1CCC(NC(c2cccc(F)c2F)=O)C1 C1(CC(=O)NCC(C)CC2CCC2)CCCC1NC(c1ccncc1)=O N1(C(c2ccc(SCC#N)cc2)=O)CCC2CCCC12CNC(=O)CSC(F)F c1(CNC(C(C)Cc2ccco2)=O)cccc(O)c1F.C12(CCCCC1)C(=O)N2 N1(C(CCc2onc(CCC)n2)=O)CCCC(C)(C)C1CNC(c1nncs1)=O c1(OC)ccc([N+](=O)[O-])c(CS(=O)(=O)Cc2c(F)cc(Cl)cc2Cl)c1 CN1CCC(NC(=O)C(=O)N(CCO)Cc2ccoc2)C1(C)C CC1CC(CNC(c2ccnc(O)c2)=O)CCN1C(=O)CCc1ccccc1F Cc1ncn(-c2ccc(C(=O)OCCCCCF)cc2)c(=O)c1C c1(C(=O)NC2(CN(C(C(CC=C)CC)=O)C)CC2)ccc2c(c1)CCCC2 c1(C(N2CC3CCCC3C2)=O)ccc(S(=O)(=O)NC2CC3NCCOC23)cc1 c1(C(=O)NC2CCN(C(c3ccc(CC)s3)=O)CC2C)cn2c(n1)CC(OC)CC2 N1(C(COCC=C)=O)CCC(F)C(NC(=O)CSc2ccccc2Cl)C1 N1(C(C(CCC)CC)=O)CCc2ccccc2C(N(C)C(c2cnc(C)s2)=O)C1 N1(C(CC(CC)(F)F)=O)CC(C)CN(C(c2ccc3c(c2)CCN3)=O)CC1C CCC(CC(=O)NCCC1(NC(=O)C(C)=C2CCCC2)CC1)CC(F)(F)F C(=O)(C(C)CNC(=O)N(C(c1n[nH]c(C)n1)Cc1ccccc1)C)NC Cc1cc2[nH]c(C(=O)NC3CCN(C(=O)CC4CCC(=O)C4)C3(C)C)cc2o1 n1(C2CCCN(C3C(C)(Br)C3)C2)nccc1[N+](=O)[O-] c1(C(=O)NC2CC(C)(NC(=O)CCc3nncs3)C2)sc2cc(F)ccc2c1Cl c1(SC)cc(CN2CC(NS(=O)(=O)CCCCl)C2)ccn1 C#CCCCC(C)C(=O)NCC(CCNC(C1(COC)CCOCC1)=O)OC CC(C)(CN1CCCCC1)C(=O)NCC1CCCN1C(C1CC(=O)C1(C)C)=O c1(C(=O)NC(C2N(C(C3(CC)CCCC3)=O)CCC2)C)ccc(C)c(Cl)c1 C(C(=O)NC1CC(O)C1)(C(C)(C)C)N(C)Cc1cn(C2CCCC2O)nn1 C=CC1(NC(=NCCc2c(F)cccc2Cl)NCC2COCCO2)CCOCC1 CN1CCC(C)(CNC(c2cc(CNC(c3nocc3Cl)=O)no2)=O)C1 C1(C=O)CCCN(C(=O)C(CN(C)C)C(C)C)CC1.C1(CC(C)C)(COC)CC1 Cc1nc(Cn2cc(COCC3CN(C(=O)COCCO)C3)nn2)c(=O)[nH]c1C c1(C(N(C2CC(NC(C3C(CC)CCO3)=O)C2)C)=O)cccc(F)c1 c1(C(=O)OCC2CCN(C(C3CCC(=O)NC3)=O)CC2)cccnc1NC(C)C CCCC(C(=O)N1CCC(NC(C2CC3(CC3)C2)=O)C1C)S(N)(=O)=O CC#CCCCC(=O)N1CCC(C(=O)NC2(CO)CCSC2)C1C1CC1 N1(C(CNC(CCCCC)=O)=O)Cc2ccc(CNC(=O)C(=O)NCC)cc2C1 C(CCC(=O)NC1CC(CC(N2CCC(c3cc[nH]n3)C2)=O)C1)C1C(C)C1 c1(C(=O)NCC2OCCCN(C(C3CCC(CC)O3)=O)C2)cc2ccccn2c1 C1(NC(c2ccc(Cl)s2)=O)CCN(C(=O)C(c2ccc(F)cc2F)=O)C12CC2 C(CC(C(C)(C)C)NC(C1CCC1)=O)N(C)C(c1ncoc1-c1cnn(C)c1)=O Cc1cc(C(N2CC(O)(C3CCCN3C(C3C4CCCC34)=O)C2)=O)cn1C Cn1nc(O)cc1C(N1CC=CC1CNC(=O)C(F)(F)c1nccn1C)=O CC(C)C(C)(Cc1ccccc1)NC(=O)NC1CC(C)(C)CN1 c1(CC(=O)NCCCN(C(C(CCC)=CCC)=O)C(C)C)cccc(Cl)c1F N1(C(c2c(CCC)cccc2)=O)CC2(CC(NC(=O)CS(N)(=O)=O)CO2)C1 Cc1cc(NNC(=O)OC(c2cccc(OC(F)(F)F)c2)C)ccc1F c1(C(=O)NCC2(CNC(Cn3c(C)ncc3)=O)CC2)nc(C#N)cs1.C1(C)C(=O)N1 C1(OC(=O)CCC)CCCC1C(C(=O)OC(CC)C1CCC1)C c1(C(=O)NCCC(C)NC(c2c(C)onc2)=O)cc2c(Cl)nccc2s1 CC(C)CC(C(=O)NCCC(C)(C)CNC(C1CC2COCC(C1)C2)=O)C(N)=O n1(C(C)(C)C)cnc(C(=O)NC2CCC2NC(=O)C=C2CCSCC2)c1 C(=O)(CC(C)(C)N(C)C(c1cnsc1)=O)NCC(CC)OC N1(C2C3(C2)C(=O)NC3)CCCC(C)CC1.C=CC1CC1C(=O)OCC.C(F)(F)F C1(C(N2CC(C(C)NC(c3cnc(C)o3)=O)OCC2)=O)CC(S(C)(=O)=O)C1 Cc1ccc2nonc2c1C(=O)OCC(c1ccccc1Br)F C(CNC(=O)CCCOC(C)(C)C)(CC(=O)NC1CCOCC1O)OC C1(CNC(c2cnc3n2CCCC3)=O)CN(C(=O)CC(F)(F)Cl)C2COCC2O1 C1(NC(C(C)=CC)=O)CCCC(NC(c2sc(C)cc2N2CCCC2)=O)CC1 C1(C)(C(N2CC(CC=C)(NC(=O)C=CC(C)(C)C)C2)=O)CCCNC1=O C(=O)(C(C)(C)NC(=O)CN(C)CC1CCCO1)OCC=C c1(OC)cc(C(=O)NC2CC2CNC(=O)C(C)OC2CCCC2)sc1Br C(=O)(CC(C)(C)C)N(C1CCCN(C(c2sccc2OC(F)F)=O)C1)CC Cc1oc(C)c(C(N2C(C(=O)Nn3cnnc3)CCC2C)=O)c1C C(C)(CCCCNC(c1sccc1CC#N)=O)NC(C(F)=CC)=O c1(C(=O)NC2CC3(CN(C(CCC=C(C)C)=O)C3)C2)cnc2cccnn12 N1(Cc2cc(OCC)n[nH]2)C2CCCC1CC(NC(c1cc(Cl)c(Cl)s1)=O)C2 O=C1CC(C(=O)N2CCN(C(C3CCCOCC3)=O)CC2CF)=NN1 CCCCCC(CC)C(=O)NC1CCC(Oc2ncccn2)CC1 N#Cc1ccnc(N2CCN(C(C3CCC3F)=O)CC2)c1 c1(Cn2cc(C(CC)(C)O)nn2)ccccc1CNC(=O)Cc1cnn(C)c1 CC1(C(=O)NC2CN(C(=O)COCc3ccccc3Cl)C2)CCCNS1(=O)=O C1(C)(CC(=O)NC(C2(O)CN(C(C3(NCC#N)CCCC3)=O)C2)C)CCOCC1 C1(C(=O)NC(CNC(c2cc(C)c(C)[nH]2)=O)(C)C(C)C)Cc2cccc(F)c2O1 C1(CC)CN(C(C)=O)CCC1NC(=O)CCn1cc(-c2ccccc2C)nn1 c1(C(=O)NC2CN(C(c3ccc(O)nc3)=O)CC23CC3)cc2cnccc2[nH]1 Cc1cc(F)ccc1CNC1CC(C(=O)NCC=CC2CCCCC2)C1 C12(C(N(C(CC)CO)CC)=O)CC(CCO1)N(C(=O)C(F)C1CC1)C2 C(=O)(C1CCNc2cc(F)ccc21)OC(C)C(=O)Nc1cccc(Cl)c1 c1(C(=O)NCCOCCCN(C(C(C)N(C)C)=O)C)c[nH]c(Br)c1 c1(C(N2C(CNC(C(C)N(C)C)=O)COCC2)=O)cc(S(N)(=O)=O)c(Cl)o1 c1(C(C(=O)NC(CCOC)CNC(=O)C(C)(C)C2CC2)(F)F)ccc(F)cn1 N1(C(C(C(C)C)OC)=O)C2CCC1CC(NC(=O)C(C)C(C)C)C2 c1(NC(c2c[nH]ccc2=NCCN2CCCC2)=O)ncc2c(Cl)cccc2n1 C1(NC(COC)=O)C2CC3CC(C2)CC1(CNC(=O)C1CCCc2c[nH]nc21)C3 N1(C(C(=O)NCC23CCC(CC2O)C3)=O)CCCC(CO)(NC(C2CC2)=O)C1 Cn1c(C(=O)NCC2CN(C(C3Cc4nccn4C3)=O)CC2O)ccc1C#N c1(CNC(c2c(C)n(C)nc2)=O)ccc2c(c1)CCN(C(C1CC(C)CO1)=O)C2 C1(C(N2CCC(OCCNC(CCOCC#C)=O)C2)=O)CCC(C(C)C)CC1 C1(C(=O)NC(C)(C)CCNC(c2cccc(=O)o2)=O)Cc2nccn2C1 C(=O)(C1CCCn2nccc21)N1CCCC2(CN(C(C3=CCCC3C)=O)C2)C1 N1(C(C(c2cccnc2)OC)=O)CC(CNC(=O)CC(C)(C)C)OC2(CCC2)C1 Cc1c(C(=O)NCC2CC2NC(c2cc(C3(C)CC3)on2)=O)ccc2cncn12 C1(NC(C(CC)n2cncn2)=O)CC2(C1)CN(C(=O)CC(C)C(F)F)C2 Cc1nc2cccc(C(N3CCCC3CNC(c3ccncc3F)=O)=O)c2[nH]1 C(=O)(C1CCC(=O)c2cccn21)N1C(CNC(c2cc(Cl)c[nH]2)=O)CCC1 c1(N2CC3(C(C(=O)OC)CN(C(C(C#C)(C)C)=O)C3)C2)ccc2c(n1)CCCC2=O N1(C(c2ccnc(OC)n2)=O)CCC(NC(=O)CCCC(F)(F)F)CC(O)C1 S(=O)(=O)(CC1CCCc2ccccc21)N1CC(C(c2n(C)ccn2)C(F)(F)F)C1 C1(C(N2CC(CNC(c3cnco3)=O)OCCC2)=O)CC2CCC1C21CC1 C1(C(=O)NCCN(CCC)C(c2nscc2N)=O)CCCCC1C Cn1nc(C(=O)NCC2CC(NC(C3CC4(C3)CC4F)=O)C2)c2c1CCC2 c1(CNCC(N2CCNCC2)=O)c(C(F)(F)F)cccc1F N12CCOC(C1)CC(=O)N(C)C1CC(C1)C2=O.C1CCC2(CC2)C1.CCO n1(CC)cc(C(=O)NCC2CCN2C(c2cc(F)n(C)n2)=O)c2ccccc12 N1(C(C2CCC(NC(C3(C)C=CCCC3)=O)CC2)=O)CC2(CCOC2=O)C1 c1(NC(CC2(CNC(c3cnc(CC)o3)=O)CC2)=O)ccc(C)nc1CC c1(N(C)CC2CCCN(C(C(c3c(C)cccc3)C)=O)C2)nc(C)ncc1C c1(C(C2CC2)NC(=O)C(N2CCC(C(C)NC(=O)OC)C2)(C)C)ncccc1C CC(C(=O)OC(C)(C)C)C(=O)NCCN(C(C1(C(C)(C)O)CCC1)=O)C1CC1 c1(CSCC)cc(C(=O)NCC2CC2NC(=O)C=C(CC)CC)c(C)o1 C(CCSC)(C(=O)NC1(C(=O)NCCC)CCC1)NC(CCOCC#C)=O Cc1cn2c(n1)CC(C(=O)NC1CCCCC1N(C)C(C1C(C)C1C)=O)C2 N1(C(c2c(C)ccc(N(C)C)c2)=O)CCN(C(C2CCCN2)=O)CCC1C c1(C(=O)OC(c2nc(C)oc2C)C)cc(Br)cc(F)c1F n1(CCCC)nnnc1C(C)(CC1CCCCC1)NC(C)C.N12CCCC1C2=O N1(C(c2c(Cn3cc(C(C(C)C)O)nn3)cccc2)=O)CC2CCCC(C1)N2C S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)NC1CN(C(C(C)(C)OC)=O)CC1C C1(C(=O)NCCCNC(c2sccc2Cl)=O)CCCC2(C1)CC2(F)F c1(C(=O)NC(CNC(CC(C)OC)=O)C(C)(C)C)oc2ccccc2c1Br CCCC(C)(O)CC(=O)N1CC(C(=O)NCc2cnc(C)s2)C(C2CC2)C1 N12CCC(C(O)C1)CNC(=O)C2=O.c1(CC)csc(SC)c1CC(C)C N1(C(C(C)S)=O)CCC2(CCN(C(c3cccc(-c4ccncc4)c3)=O)C2)C1 C1(NC(C2(S(N)(=O)=O)CCCC2)=O)CC2CCC1CN(C(C1CC(=O)CO1)=O)C2 C1(=O)C2=CCC(C2)N1.c1(COC)cc(C)c(C(=O)O)o1 C(c1ccccc1Cl)=CC(=O)N(CC(C)NC(C(C)CC1CCCO1)=O)C C(=O)(N=c1cc2ccccn2[nH]1)C1C(C)(C)C1CNC(=O)Cn1nccn1 C(C1CCCN1C(=O)C(C)CC#N)=CC(=O)NC(C(=O)OC)CO C1(C(F)(F)F)(NC(C2C(C(CO)NC(=O)CN3CCCC3=O)C2)=O)CCCC1 Cc1ccc(C(C)C)c(-n2cc(CNC(C3OCCN(C)C3=O)=O)nn2)c1 c1(N)ccc(C=O)cc1.C1(N(CCOC=O)CC)CCN(C2CCOCC2)C1 c1(C(=O)NC(C2CN(C(c3cc(C#N)on3)=O)CCO2)C)ccc(F)c(Cl)c1F CCC(CC)C(C)C(=O)NC(CC)CCCC(=O)NCCCOC(F)(F)F CC(C)C(C(=O)NC(C(=O)NCCC1(O)CCOC1)C1(C)CC1)C(C)C C(=O)(C(C)(C)CC(F)F)NCCCC(C)NC(C(C)CSC(F)(F)F)=O c1(OC)cc(OC)cc(CCC(=O)NCC2CCN(C(=O)C(Cl)=CCl)CC2C)c1 CC1(NC(C2CCCC(F)(F)C2)=O)CCN(C(=O)C2=CCCCO2)CC1 c1(C(N2CCN(C(CSC)=O)CC2c2cn[nH]c2)=O)cnc2ccc(C)cn12 C1(C(N2CCC(CNC(c3cc(CCC)on3)=O)C2)=O)CCN(C2CC2)S1(=O)=O C1(CNC(C=CC)=O)CN(C(c2cc(OC)nc(Cl)c2)=O)C(C)(C)C1 C1(NC(CC2CCC(C)CO2)=O)CCSC12CN(C(C1(CO)CC(F)(F)C1)=O)C2 C1(C(N2CCCC(CC(N)=O)C2)C(=O)NCC(C)C)CCCC(C)C1 N1(C(c2cc(OCC)ncc2)=O)C2CCC1CC(NC(c1cc3ncsc3[nH]1)=O)C2 c1(CNC(C2(C#C)CC2C2CCN(C(=O)OC(C)C)C2)=O)cccc(C)c1 Cc1c(-c2csc(Nc3cccc4sccc34)n2)oc2ccccc12 N1(C(C=Cc2c(C)ncs2)=O)CCCC(F)(CNC(c2coc(N(C)C)n2)=O)C1 N1(CC(CSC(C)(C)C)=O)CCC(NC(=O)NCCOc2ccc(F)cc2)CC1 N1(C(=O)COCCN(C)C)CCC2(NC(C3CCCCCC3)=O)CCCCCC12 c1(C(N(CC(C)CNC(=O)CCc2cc[nH]n2)C)=O)cc2c(O)ncnc2cn1 C1(NC(CC2(C)CC2)=O)CC12CCN(C(=O)COC(=O)CO)C2 C#CCC(C)(CC)C(=O)NCC1CN(C(c2cnn(CCOCC)c2)=O)CCO1 CCC(CC#N)N=c1[nH]c(=NC(C)c2n[nH]c(C(C)C)n2)[nH]c2ccsc12 C1(C(=O)NCc2c(CCNC(CSCCC)=O)ocn2)C2CCC1CC2 c1(C(=O)NCC2N(C(C(C)CO)=O)CC(O)C2)ccc2c(=N)[nH]cnc2c1 C(=O)(C(CCC1CC1)NC(=O)C=CC1CCC1)N(C)Cc1ccoc1 N1(C(c2cnc(CO)cn2)=O)CC(CNC(C2(CO)CCCO2)=O)CC12CCC2 c1(OC)ccccc1C(CNC(C1(C)CC(F)(F)C1)=O)NC(c1ccccn1)=O c1(C(N2CC(NC(c3cc(CO)[nH]n3)=O)(CO)C2)=O)csc2ccncc12 C1(C(=O)NCCCNC(C23OCC(CC)(C2)C3)=O)Cc2cc(C)ccc2S1 N1(C(CN2CCN(C)CC2)=O)CCOC2(CCN(C(=O)CC(C)(C)N(C)C)C2)C1 c1(C(=O)NCCCCN(C(C(c2c(C)cccc2)C)=O)C)c(Cl)nn(C)c1C C1(N(C(C2N(C(C(C)OCC3CC3)=O)CC2)=O)C)CCN(CCF)C1 C(CNC(=O)C1CC1)(C(=O)NC1CN(CC(F)F)C1)N(C)C c1(C(=O)NC2(CCNC(c3c(C)nc(C4CC4)o3)=O)CC2)cnn2c1CCC2 c1(C(=O)NCCC(C)N(C(C2C(C)(C(C)C)C2)=O)C)cccn2cnnc12 CCCC(CCCO)C(=O)N1CC2CC1C2NC(=O)CCn1nc(C)cc1C N1(C(COCCC)=O)CCC2(CCCC2NC(c2c[nH]c3ccc(C)cc23)=O)C1 c1(N(CC(=O)NCc2nccn2C)C)nc(=NCC2CCCCO2)[nH]c2ccsc12 c1(C2C(C=O)C2)ccc(Cl)c(Cl)c1.N1(CC=O)CCCCCC1.N12CC(C1)N2C Cc1cc(C(=O)NC(c2ccc(F)cc2)(C)C)cc2ccccc12 N1(C(c2c(CC)cc[nH]2)=O)CCC(C)(C)CC1C(=O)N(C1CCOC1=O)C C(C1CCCC1)=C(C)C(=O)NC1CC1NC(=O)CC(=O)NCC1CC1 Cc1cc(C(=O)NC2CCCCC2NC(c2cnnc(C)c2)=O)n(C(C)(C)C)n1 c1(C(=O)NC2C(CNC(c3cnc4[nH]nnc4c3)=O)C2)scc2c1OCCO2 N1(C(C(COC)(C)C)=O)CCC2(NC(c3cncc(-n4cnnn4)c3)=O)CC2C1 N#Cc1cccc2[nH]cc(C(=O)NC3CCCC3CNC(=O)C(Cl)=CCl)c12 N1(C(C(CC)SC)=O)CCN(C(=O)CCc2ccn(C)n2)C(CF)C1 c1(OC)ccnc(O)c1C(=O)NC1CC(NC(c2ccc(SC(F)F)cc2)=O)C1 c1(C(CNC(c2cc(O)cs2)=O)NC(C2C(C)(C(C)C)C2)=O)ccccc1 c1(NC(C2CN(C(=O)CNC(C3CC(CF)C3)=O)C2)C)ccc(Cl)s1.C1CC1 C1(NC(c2cc(CCC)on2)=O)CN(C(=O)C2=NOC(C)C2)C(CC)(CC)C1 N1(C(C=CCCCCC)=O)CCCCC1C1CCCN1C(=O)Cc1cc[nH]n1 N1(C(N)=O)CCCC(C(=O)NCCNC(=O)C(CO)c2ccccc2)C1 c1(Cn2c(C)nc(-c3nc(C4CC4)nn3C)n2)ccc2ccccc2c1 c1(CNC(C(C2CCOC2)OC)=O)nccn1C(F)F Cc1cccc(O)c1C(=O)NC(C)C(C)NC(c1ccsc1C#N)=O Cc1oncc1C(=O)NCC1CC(NC(=O)CCOCC(C)C)C1 CN1CCN(C(c2cnn(CCNC(=O)C=C3CCOCC3)c2)=O)C(COC)C1 CCCC(C)CCCC(=O)NCC1(CNC(=O)CCSCC)CC1 CCC(C)C(C(=O)NCCC(=O)NC(c1cn(C)nc1C)C)OC C1(CNC(c2nc(CC)oc2)=O)CCCN(C(=O)CSc2ccc(Cl)cc2)CC1 N1(C(C(C)=CC)=O)CCN(C(c2c(C)ccc(C)c2O)=O)CCC1C C#Cc1cc(C(=O)N(C2CN(C(c3cnnn3C)=O)CC2F)C)cc(F)c1 S(=O)(=O)(CCC(=O)N1CC(O)CC1CC1CCCOC1)NC(=O)OC(C)(C)C S(=O)(=O)(c1cccc(S(=O)(=O)N2CCC(c3cccnc3)C2)c1)N(C)C c1(CC)cc(C(=O)NCC2CCN(C(=O)C(C)(C)C(N)=O)CC2C)ccc1Cl C1(CCNC(C2CC23CC3)=O)CN(C(=O)CNC(c2ccsc2)=O)CCS1(=O)=O N1(C(CC(C)N2CCCC2=O)=O)CC=C(CNC(=O)CC2(C)CC2(Cl)Cl)CC1 C(C(=O)NCC(C1CC1)NC(C1C(c2nc(C)no2)C1(C)C)=O)(C(C)(C)C)SC c1(C2(NC(=O)Nc3cccnc3Cl)CC2)ccc2c(c1)OCCO2 CC1=C(C(=O)NCC2CN(C(=O)CS(=O)(=O)NC3CC3)CC2C)CCC1 Cc1cc(C(N2CCCC2(C)CNC(c2cc(C(F)F)ncn2)=O)=O)cnc1O c1(OC)ncnc(C)c1C(=O)NC1CC1NC(C1CC(=O)N(C)C1)=O C#CCC(C)(C(=O)NCC1(CCO)CC1)NC(=O)C(C(C)C)N(C)C N1(C(C(=O)Cc2ccccc2)=O)CCC2(CCC2C(=O)Nc2ccccc2)CC1 c1(CNC(=O)CCNC(C2(CNC(=O)CC3COC(=O)C3)CC2)=O)ccccc1 C(=O)(CC1=NN(C)C(=O)C1)N(CCN(C(c1cc(C(C)C)nn1C)=O)C)C(C)C Cc1ccc(C(=O)NCC2COCCN2C(=O)CC2(N(C)C)CCC2)c(C(N)=O)c1 C#CCC(CC#C)C(=O)NCC1CN(C(c2cccc(C(F)F)c2F)=O)CC1C C(=O)(C(C)(C)CC(F)F)NCC1(NC(c2cnc(CC)nc2C)=O)CC1 C1(NC(CSCC)=O)CC(NC(=O)CSCC(=O)NC)C1 N1(C(C(CC)=CCCC)=O)CCC(CN(C(=O)C(=O)NCCOCCOC)C)CC1 C1(C(C(=O)NC2(COC)CC2)C)CCCN(C(=O)COC(C)(C)CSC)C1 C(=O)(C(F)C(C)CNC(=O)Cc1ncoc1C)N1CC(OCC)C1 C(=O)(C(F)C(C)(C)O)NC(CCCCNC(C(c1ccc(C)o1)C)=O)C N1(C(C2(C(CC)=O)CC2)=O)CCC(C(N2CC(OCC)C(F)C2)=O)C1C N1(C(C(C)(C)NC(=O)OC)=O)CC(NC(=O)C(O)CCSC2CC2)C(C2CC2)C1 CC(CC(=O)NC1CC2CC(NC(=O)C(C)(C)N3CCOCC3)C2C1)C(F)F O=C(C1=CCCN(C(=O)CC2CCCO2)C1)NCc1cc(C2CC2)on1 c1(C(=O)NC2(C)CN(C(C(CC)(C)CC)=O)C2)ccc2c(N)nccc2c1 C(=O)(C1=C(Cl)CCC1)N1CC(CC=C)(NC(c2cccnn2)=O)C1 C1(CNC(=O)C(=O)OC(=O)Cc2ccc(F)nc2)CCCC2CNCC12 c1(C(N2C(C)CC(NC(=O)CSc3nncs3)CC2)=O)snc2ccccc12 N1(C(c2scc(C)c2)=O)CCCCC1C(C)(C)CNC(c1cc(Cl)c[nH]1)=O N1(C(c2ncc(NC)nc2)=O)CC(NC(c2cc(C)on2)=O)CC(O)C1 C(CC)(CCC(=O)NCc1cccs1)NC(c1c(NC)cccc1)=O C(=O)(C(C)(C)CC1CCOCC1)NC(C1CCN(C(=O)Cn2cccn2)C1)C C(CC(CC)C(=O)N1CC(O)CC1(C)C(=O)Nc1cc(CC)cc(O)c1)=CC N1(c2cc(N3CCC4CCC(SC)C43)nc(C)n2)CC(C)(C)OC(C)(C)C1 N1(CCC(=O)NC(CC=C)CNC(=O)CC2CC(=O)C2)CCCCC1=O c1(CCCC(=O)NC2(C)CN(C(C(CC)SC)=O)C2)cccc([N+](=O)[O-])c1 C1(c2nnnn2C(C)C)(NCc2cc(OC)c3c(c2)OCO3)CC2CC1CC2F c1(-c2ccc(OCC)nc2C)cccc2c(C(=O)Nc3nc(C#N)cs3)[nH]nc12 C(=O)(C(C)(C)CC1CC1)NCCC1N(C(C=CCN(CC)CC)=O)CCC1 N1(C(CC2ON=C(C)C2)=O)CC(NC(c2cn3cccnc3n2)=O)C2(CCC2)C1 CCCCCCCN(C(=O)C(Cc1cnc[nH]1)NC(c1cc(O)nn1C)=O)C N1(C(C(CC)OC)=O)CC(CNC(c2nn(C)cc2C)=O)OC2COCC12 O=C(CC(O)C1CCCC1)NCc1c[nH]nc1C(=O)NC1CC(C(F)(F)F)C1 C1(c2ccccc2)(CNCCC(C)OCC=C)CCN(C(=O)OC(C)(C)C)CC1 C1(CNC(C(COCC)(C)C)=O)CC2(CO1)CN(C(=O)CCCN(C)C(C)C)C2 C12(C(=O)NCCC3N(C(C(CC#C)C4CC4)=O)CCC3)CCC(CC1)C(C)O2 CC1C2C(CCN2C(=O)CC2CCSC2)CN1C(C1CCCC1)=O C1(NC(C(C(CC)C)O)=O)COC2(C1)CN(C(c1csc3nnsc13)=O)C2 N1(C(CCC(C)NC(C=CC=CCC)=O)=O)CCC(C)C(CO)C1 c1(OCCNC(=O)NC23C(C)(C)C(C2)C3)ccc(C#N)cc1 Cc1cccc(C(=O)NC(C)CCCNC(c2nc[nH]c2C(F)(F)F)=O)c1Cl c1(C(n2cc(CNC(c3c(C)cc(CC)o3)=O)nn2)(C)C)ccnc2[nH]ccc12 c1(N2CCC(COC)(NC(C3CC3(C)Br)=O)CC2)c(C)cccc1[N+](=O)[O-] C1(CNC(c2c(C3(C)COC3)noc2)=O)CC2(CCOC2)CO1 N1(C(CC(=C)C)=O)CC(NC(c2cc(-c3ccccc3F)[nH]n2)=O)C2CC2C1 c1(OC)ccnc(O)c1C(=O)NCCC(C(C)C)NC(c1cnn2c1OCC2)=O C1(CC(=O)OC)C(=O)NCCN1Cc1ccc(-c2ccco2)s1 c1(NCC(=O)NCCOC)ccc(S(=O)(=O)NCC2CCOC2)cc1F CCCC(C)(O)CC(=O)N(CCNC(c1cncc(C(F)(F)F)c1)=O)C1CC1 c1(OCC(N2CCC(NC(C3(C#C)CCC3)=O)C2C)=O)cc(Cl)ccc1Cl C1(CC)CN(C(=O)C(C)SC)CCC1NC(c1cccc(Cl)c1OC)=O N1(C(CCNC(=O)NC)=O)CC(CNC(C2CC2(C)OC)=O)CC12CCOCC2 N1(C(c2nnn(C(C)(C)C)n2)=O)CC2(C1)CN(C(=O)C(C)(C)n1cnnn1)CCO2 c1(CN(C(C(c2ccco2)NC(c2ccc(C)s2)=O)=O)C)c(C)noc1C C(F)(C(=O)NOC1CCCCC1)C1CC(N2CC(C)(OC)C2)C1 C(CC(=O)Nc1nc(C(F)(F)F)cs1)(C(F)F)NC(c1n(CCOC)ncc1)=O c1(C(=O)NCC2CC(F)(CNC(c3ccc(C(N)=O)s3)=O)C2)cc(O)nc(Cl)c1 C1(NC(N2CCN(CCN3CCOC3=O)CC2)=O)CCC(C2CC2)C1 c1(C(COC)=O)cccc2c(CCn3nc(C)cc3C)cccc12 N1(C(=O)OC(C)(C)C)CC(NC2CCCC2)C(CC(C)(C)C)C1 N1(C(C2CC(OC)(OC)C2)=O)CCC2(CC(NC(=O)CSCCC(C)C)C2)C1 Cc1ccnc(C(N2CC(NC(=O)C(C(C)C)C3CCC3)C(F)C2)=O)c1F c1(C(N2CCC(N(C(C)C)CC)CC2)=O)cccc2nc(C(Cl)Cl)[nH]c12 c1(C(=O)OC)ccc(C(=O)NCCCC(C)NC(=O)CC2CC23CC3)cn1 C1(NC(c2csnc2Br)=O)(CO)CN(C(=O)C(C2CCCCC2)O)C1 N1(CCO)CCN(C(=O)C=CCF)CC1.CC(O)C(=O)N c1(C(N2CCCCC(NC(C3N(C)CC(F)C3)=O)C2)=O)cc(S(N)(=O)=O)cn1C N1(C(c2c(C)oc(CO)c2)=O)CC2CC(C)N(C(=O)CC3CC(C)(C)CO3)C2C1 N1(C(c2cc(OC)n3c2COCC3)=O)CC(=O)Nc2c(C)ccnc21.CO c1(CNC(=O)NCCOCC#C)cnc(O)c(Oc2ccc(OC)cc2)c1 c1(OC(C)C(N2CCOC(CNC(C3(O)CCOCC3)=O)C2)=O)cccc(F)c1 C1(CC(C)NC(c2n(CC)ncc2)=O)CCN(C(C2CC2C#N)=O)CC1 C1(C(=O)NCCN2CCN(C(C=CC)=O)CC2)CCC(=O)N2CCCC12 CCCC(C(C)C)(c1nnnn1C(C)(C)C)NC(C)CC(C)OC N1(C(c2ccncc2)=O)CC(F)(C(N2CCC(OC3CCC3)C2)=O)C1 C1(C(=O)NCC2ON=C(C(C)C)C2)Cc2cc(Br)ccc2O1 C1(C(=O)NCC2N(C(CC3(C)CCC3)=O)CC2)CCC2(CCCC2)C1 CC1CN(C(c2cc(C(N)=O)[nH]n2)=O)CCN1C(=O)Cc1nncn1C CN1CCC(C)(C(=O)NCC(C(=O)NC2CCC3(CC3)C2)N(C)C)CC1 C(=O)(C(C)CC(F)(F)F)N1C(Cn2cc(C3CN(C(CC=C)=O)C3)nn2)CCC1 O=C(CC(F)(F)c1ncc[nH]1)Nc1ccc(Oc2nc[nH]n2)cc1 N1(C(c2c(C)cc(C)[nH]2)=O)CC2ON=C(CNC(=O)Cc3nocc3C)C2C1 C(=O)(C(COC(=O)N)Nc1ccccc1)OC.C(C=CCl)OC(C)=O N1(Cc2ccc(CC(=O)OC)cc2)CC2(CCC2)C1CC1CC1 c1(CC)cccnc1C(=O)NC(CNC(C1COCCN1CC1CCC1)=O)CC c1(OCC)cc(CC(=O)N(CC(C)NC(C2(CC)CCCC2)=O)C)ccn1 N1(S(C(C)C)(=O)=O)CC2(CN(C(C3CC3F)=O)CCO2)C1 c1(C(=O)NC2C(C)CN(C(=O)CC#N)CC2)ccnc2cc[nH]c12 C12(C(N3CCN(C(C(C)CC(N)=O)=O)CC3CF)=O)CC3CC(C(=O)N1)C2C3 C1(NC(c2c(CCC)onc2C)=O)CC2CCC1N(C(=O)C(C)n1cccc1)C2 C(=O)(C1=NOC(C)(C)C1)NC1C(C(=O)NC(CC(CC)C)CO)OCC1 c1(C2(C(=O)NCC(C)NC(=O)COc3ccccc3)CC2)ccc(F)cc1Cl.C1(C)CC1 C(CC(C)C(=O)NC(c1nocc1C(=O)NOCC1CCCO1)C)=CCC c1(OCC)ccc(C)cc1C(=O)NC1(COC)CN(C(C2CCC2(C)C)=O)C1 N1(C(C(C)CC2CCC2)=O)C2CCCC1CC(NC(c1ccc(F)c(O)c1)=O)C2 c1(C(=O)NCC(=C)CCNC(=O)C(O)P(C)(C)=O)cc2ccc(OC)cc2cn1 C#CCCCCC(=O)NC1CCOCC1C(N1CCC(F)(C(N)=O)C1)=O C1(C(C)(C)C)CCC(N=c2ccc3c(F)ccc(F)c3[nH]2)C(=O)O1 C(=O)(CCCCCO)N1CCC(NC(CC2(C)CCOCC2)=O)C1(C)C CC1CN(C(=O)COCC(C)(C)C)CCCN1C(=O)CNS(=O)(=O)c1cccs1 Cc1cc(C(=O)NC2(C)CC=CCC2)c2[nH]cnc2c1 C(C(CC(C)C)C(=O)N1CC2CC2C1C(=O)NC(C)CCC=C(C)C)OC c1(NCc2cnc(CC)s2)ccc(S(=O)(=O)N2CCCCC2CCO)cn1 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 Cc1oc2cc(C(=O)NCC3CC(CNC(c4ccncn4)=O)CO3)[nH]c2c1C [N-]=[N+]=NC1CCN(C(C2CN(C(c3ncc(F)cc3F)=O)CC2(F)F)=O)C1 C1(CNC(C=C(CC)C)=O)CC2(CCC2)CN1C(c1cnc(CC)nc1)=O C=C(F)C1(CC(=O)NC(CNC(=O)CC2CCCOC2)CCCC)CCOCC1 c1(NC(=O)CCCn2cc(C3COCCOC3)nn2)ccc2[nH]ccc2c1 CCC(C)(COC)C(=O)NC1CS(=O)(=O)CC1NC(c1ccccc1Cl)=O C(C)(CN=c1[nH]cnc2cccc([N+](=O)[O-])c12)(C1CC1)NC(C1C(C)(C)CC1)=O N1(C(C(C)=O)=O)CC(NC(=O)C=CC(=O)N(C)C)CC12CCOCC2 C(=O)(C#CC1(C)COC1)N(C)CCNC(c1ccn2c1CSCC2)=O N1(C(=O)Nc2cccc(C(F)(F)F)c2)CC(F)CCC(F)C1 c1(OC)cc(OC)c(C(N2CCC(CNC(c3csnc3C)=O)C2)=O)cc1Br C1(C(=O)NCC2C(OC)(OC)CC2)CCNCC(C)(C)C1 C12(C(N3C(CC(N)=O)CCC3)=O)COC(C1)C(NC(=O)CN1C=CC1(F)F)C2 c1(OC(C(=O)NCC2N(C(C(COC)OC)=O)CCC2C)C)ccc(F)c(F)c1 c1(C(N2CC(CC(C)NC(C=CCC)=O)C2)=O)cc(Cl)cc2c1OCC2 c1(CC2CN(C(C(Cc3cn(CC(CSC)(C)C)nn3)C)=O)C2)ccccc1Br c1(C(N(C)Cc2ccc(C)cc2Cl)=O)cc(C#N)c(F)c(F)c1F S(=O)(=O)(c1cccnc1Cl)N1CC2(CN(C(=O)CO)C2)C1 C(=O)(C1=C(C)CCOC1)NC(CC(=C)C)C(=O)NCC(C)(O)C(C)C c1(SC(C(=O)NCCN(C(CCOCC)=O)CC)C)nncn1C C(=O)(C(CC(C)(C)C)OC)NCC=CC.c1(C2C(=O)N2)ccnn1C c1(C(=O)NCCC(C)NC(Cc2cc(C)[nH]n2)=O)ccnc2c1nnn2C C=CCC(F)(F)C(=O)NC(CC)CC(=O)N1CCCC(OC2CC2)C1 C(=O)(CCCn1ccnc1)NC(CN(C(c1ccsc1C)=O)CC)C c1(OC)ccc(C(N2CCCOC(CCNC(c3cscn3)=O)C2)=O)c(C)n1 CC(C)CC(F)(F)C(=O)NCC1CCN(C(=O)C(F)OC(F)(F)F)CC1 C(=O)(C(F)(F)C(O)C1CC1)NCC(C)(CNC(C1C2CCN1CC2)=O)OC Cc1nccc(C(=O)NCC2CC(C)(C)CN2C(=O)C(O)P(C)(C)=O)c1C Cc1cc(C)c(C(=O)NC2CCCC2C(=O)NCc2ccc(F)cc2O)cn1 C1(CC(NOCC)=O)(Nc2cc(C(F)(F)F)n[nH]2)CC2CC2C1 C(=O)(CCS(C)(=O)=O)N1CC(C(N2C(C)CC(F)C2)=O)C(C)C1 N1(C(c2cc(C(C)C)no2)=O)CCC2(CCN(C(=O)CC3(CO)CC3)C2)C1 c1(C(=O)NCCC(C)N(C(c2ncn(C(C)C)n2)=O)C)cc(O)cc(Br)c1 C1(C(=O)NCC(CC=C)NC(c2ccc(Cl)cc2CC)=O)CCCCN1N=O CCCCC(CC)CCC(=O)NCC(c1ccc(C)cc1)NC(=O)C(O)C(C)C c1(C(N(CCCNC(CC2(C)CC2F)=O)C2CC2)=O)c[nH]nc1-c1ccc(Cl)s1 Cc1[nH]nc(C(N2CCC(NC(=O)CCN3CCN(C(C)C)CC3)C2C)=O)c1C CC1CN(C(=O)CN2CC(=O)N(C)C2=O)CCC1NC(c1cc(Cl)nnc1O)=O CC(C)C(C(=O)NCCCC(C)(C)NC(=O)CN(C)C)n1cncn1 c1(CCC)nnc(S)n1CC(=O)NCC(C1CC1)NC(c1cnc(C2CC2)[nH]1)=O C(C(N=c1nc2ncn(C)c2c(NC2CC2)[nH]1)C1CCC1)NC(CCC(=O)NC)=O C1(C(=O)NC(C)CNC(c2ccn(Cc3ccccc3)n2)=O)COC(C)(C)CO1 c1(N2CC(C(=O)NC3CC(C)N(C(=O)C(C)(C)C)C3)C2)nc2ncccn2n1 C1(C(N2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC2CO)=O)CCc2nccn2C1 CC(C)C1=NOC(C)(C(=O)NCCNC(=O)C(C)NC(c2ccoc2)=O)C1 C1(C(N(CC(CC)O)C)=O)(C(=O)O)CCOC(C)(C)C1 N1(CC)CCCC1C(N1CC(N(C(=O)CCOCC2CC2)C)C1)=O N1(C(c2c(SCC)nccn2)=O)CCCC(CC)(NC(=O)CN(C2CCC2)C)C1 N1(C(C2C(CC)C2)=O)CC2(C)CN(C(c3ccc(N)c(Cl)c3)=O)CC2(C)C1 N1(C(CNC(=O)Nc2ccns2)=O)CCC(NC(c2cnsc2)=O)C(F)C1 n1(CC(=O)NC2CCC2CNC(C23CC(C2)C3)=O)ccc2ccccc12 N1(C(c2c(C)oc(CO)c2)=O)CCC(NC(c2ccnc(S)c2)=O)CC(C)(C)C1 Cn1nccc1C=CC(=O)NCC12CCC(NC(=O)C=C3CC3)(C1)C2 c1(OC)c(F)ccc(C(N2CCC23CN(C(c2cc[n+]([O-])cc2)=O)C3)=O)c1F C(=O)(CC(C(F)F)NC(=O)CC=C)N1CC(CC#C)OCC1 c1(OCC)nc(C(N2CCC2CNC(C2CCCN2CC(C)C)=O)=O)co1 Cc1cccc(Oc2ccnc(N(c3ccccc3)CC(F)(F)CO)n2)c1 c1(CC)ccc(C)cc1C(N1CCCC(CNC(=O)CCF)CC1)=O c1(OCC(=O)NC2CCN(C(C3(C)CC(=C)C3)=O)CC2F)cccc([N+](=O)[O-])c1 N1(C(c2ccc(C(C)(C)C)cn2)=O)CCC2CCC(C1)N2C(C1CC(F)(F)C1)=O CCC(C)(CNC(C1CCOCC1)=O)C(=O)NCC1(CCO)CN(C)C1 N1(CC(=O)NC2CC(NC(CC3(O)CC(C)(C)OC3)=O)C2)C(=O)NC(C)(C)C1=O N1(C(CCNC(N)=O)=O)CCCOC(CNC(=O)C=CBr)C1 c1(NC(C)=O)ccccc1CC(=O)NC12CC1CN(C(=O)C=CC(N)=O)C2 c1(C(=O)NC2C(C)CN(C(=O)Cn3cccnc3=O)C2)ccc(N)c(O)c1 C(=O)(CC(C)C(C)(C)NC(=O)CCOCC(C)C)NC(c1ccncc1)CC Cn1cnc2ncnc(N3CC4(CC4C(N4C5CCCC4COC5)=O)C3)c12 N1(c2nccc(C#N)n2)CCC2(CC(C(=O)N3CC4OCC(F)(F)C4C3)=NO2)C1 CC(C)(O)CC(=O)N(CCNC(C1CCCCS1)=O)Cc1cccc(Cl)c1 c1(CN2CC(NC(=O)Cc3cc(Cl)ccn3)C(F)C2)cccc(Br)c1I N1(C(C2(COCC)CC2)=O)C2CCC1C(F)C(NC(c1nccnc1CC)=O)C2 C1(N(N2CC(Cc3n[nH]c(=N)s3)C2)C(N(C(C)C)CC)=O)CCN(C)CC1 C=CC(C)(C)CC(=O)NC1CCN(C(=O)Cc2cc(C)ccc2OC)C12CC2 c1(C(=O)NC(CN(C(=O)COC(C)C)CC)C)cccc[n+]1[O-] C(=O)(C1CCCc2n[nH]cc21)N1CC(C)SCC1.C(=O)C(C)(C)C(F)F C1(OC)CC2CC(C(=O)NCCOCCCN(C)C(c3nscc3C)=O)CC12 C(CC(C(C)(C)C)NC(=O)CCCF)N(C)C(c1cnc(O)n1C)=O C#CC1CCCC(CNC(C2CN(C(=O)C=NOC)C(C)(C)C2)=O)C1 CC1CCC(C)N1CC(N1CC(NC(C2CC23CCOC3)=O)C(C)C1)=O N1(C(CC(CC(=O)OC)C)=O)CCC2(CC1)CCN(C(c1cn[nH]c1)=O)CC2C c1(C(=O)NC(C(CO)NC(Cn2c(C)nnn2)=O)C)ccc(CC2CC2)cc1 C1(C(N(CC(=O)OC)C2CC2)=O)CCC(C2CC2)N1C(=O)Cc1cscn1 N1(C(C)C(N)=O)CCC2CCC(C1)N2C(c1cnn2ccc(O)nc12)=O N1(C(C(C)CC2CC2)=O)CC(CNC(c2cnsn2)=O)CCC1C n1(CCCC)cc(C(=O)NCC2CN(C(=O)CCOC3COC3)CCO2)c(C)n1 C(=O)(CC(C(C)OC)NC(=O)Cc1ccnn1C)N(CC)Cc1ncc[nH]1 N1(C(c2ccn(CCC)n2)=O)CCOC(CCNC(=O)CC2CNC(=O)C2)C1 CC(CNC(C1CCc2nccn2C1)=O)N=c1cc(C(N)=O)nc(Cl)[nH]1 C1(C(=O)NCCCOCC)(CNC(=O)C=CCN2CCOCC2)CCCCC1 C1(CC)CN(C(c2cn(CCCOC)nc2)C(=O)Nc2ccccc2)CC1O c1(OC(CC)C)ccc(C(=O)NCC(C)NC(=O)C(F)(F)c2csc(C)c2)cc1 Cn1cc(C(N2CCC(c3cn(CC(C)(C)O)nn3)CC2)=O)c(O)nc1=O c1(N(C)C)ccnc(C(=O)NC2CCCC2NC(c2cnc(C(F)(F)F)s2)=O)c1 Cc1nc(NC(c2cccc(Br)c2)CF)cc(=NCc2ccc(F)c(F)c2Br)[nH]1 c1(C(=O)NC(C(C)OC)C(=O)N(CCN=[N+]=[N-])C)ccc(=O)n(C)c1 C=C1CCN(C(C2CCCCC2)=O)C(C(=O)NC(c2nc(C)cs2)C)C1 C1(C)(C(=O)NCC(CN(C(c2ccnn2CCF)=O)CC)(C)C)CC(C#N)C1 Cc1cc2nc(C(=O)NC(C)CCN(C)C(c3cnns3)=O)cn2cc1C C1(F)(C(N2CCC(OCC(C)C)C2)=O)CCCN(C(=O)CC2CCSCC2)C1 C(=O)(CC(C)NC(N)=O)NCCOCCOCCC c1(OC)ncnc(C)c1C(=O)NCC(O)CCNC(C1C(C)(C)C1(C)C)=O CC1(CNC(C2CCCCC2O)=O)CCCN1C(=O)C=Cc1cccnc1 c1(C(=O)NCC(C)N(C)C(C2CCOC(C)(C)C2)=O)csc2ccccc12 c1(C(=O)NCCC2CCC(NC(c3ccc(C)n3C)=O)C2)ccc(Cl)c(F)c1N N1(C(c2n(C)ncc2C#N)=O)CC2(COC(CNC(c3cnc(Cl)cn3)=O)C2)C1 N1(C(CC2(COC)CCCC2)=O)CCC(OC2CN(C(=O)CNC(C)=O)C2)CC1 CCC(CC)CC(F)C(=O)N1CCC(C(N2CCCN3CCCC3C2)=O)C1 C12(C(=O)NCC34CC(COC)(N(C(=O)C(C)(F)F)C3)C4)CCCCC1OCC2 C1(C(=O)NC2C(NC(=O)Cc3ccsn3)CCC2)Cc2nccn2C1 CC1CN(C(c2ccc(Oc3ccccc3)o2)=O)CC1NC(=O)CN1CC=CC1 Cc1nn(C)c2ccc(C(=O)NCC3CCc4nccn4CC3)cc12 N1(C(COCCC(C)C)=O)CCCC(C)(C(N2CCCC(C)CC2)=O)C1 C(=O)(C1Cc2ccccc21)N1C(C(N2CCC(C)(O)C2)=O)COCC1 N1(C(C2N(C(C(C(=C)C)(C)O)=O)CC2)=O)CC(O)C(N=[N+]=[N-])C1 c1(C(=O)NCCCN(C)C(C2(F)CCOC2)=O)cn(C2CCOC2)nn1 N1(C(c2ccc(OC)s2)=O)C2CCC1C(F)C(NC(c1nn(C)nc1C)=O)C2 c1(CC)c(C(=O)NC2CC(CO)N(C(c3n[nH]cc3C)=O)C2)[nH]c(C)c1C(N)=O CC1(C(N2CCCC2C2(C)CC2)=O)CCN(C(c2csc(Cl)n2)=O)CC1 N1(C(C(COC)C)=O)CCN(C(c2ncoc2C)=O)CC1C C1(C)(COC)CCN(C(c2cc(C(C)(C)C)nn2C)=O)C1 C(C(CCO)NC(=O)C(C1(C)CC1)NC(c1cscn1)=O)N(C)C N1(c2ncc(C)c(C)n2)CCCC2(NC(c3ccnn3C(C)C)=O)CCCC12 CCC(CC(=O)NCC1CC(C)N(C(=O)Cn2cc(C#N)cn2)C1)CC(C)C C1(C(=O)NC(C)CCNC(=O)C(C)(C)C2CC2)CCC2(CCC2)O1 C1(C(=O)NCC2(OC)CCCC2)CC2CC2N1C(c1cccc(C2CC2)c1)=O C(=O)(CCC(=O)C(C)(C)C)NC(CCOC)C(=O)NCCC1CCCC(C)C1 C1(CC)C(C(=O)NOCCCOC)CCN1C(C1(O)CCCCC1)=O CC(C)CC(C1CC1)NC1CC1Cc1ccccc1 c1(NC(=O)C=CC=CC2CCN2)cc(C(F)F)c2cn[nH]c2c1 C(CCC(O)C(=O)NCCN1CC=CCC1)NC(C(C)CCN(C)C)=O CN1CCN(C(c2cc(O)nc(O)n2)=O)C(CNC(C23CCCN2CCC3)=O)C1 N1(C(CC2CN(C)C2)=O)CCCC2(CNC(c3cc(C4CC4)no3)=O)CCCC12 C1(NC(C(F)OC)=O)(CNC(=O)CNC(=O)COCCC(C)C)CCCCC1 c1(C(=O)NC(CN(C(C2CCC(=O)N2C)=O)CC)C)cc(Cl)cc(Cl)c1N c1(CNc2c(C)c(N3CCN(C(=O)CO)CC3)ncn2)ccc2n[nH]cc2c1 C1(CNC(C2(NC(C)=O)CCCC2)=O)CCC(C)(C)CN1C(=O)C(F)C(F)(F)F Cc1nn(C2CCC2)cc1C(=O)NC1CCC(N(C)C(c2cc[nH]c2)=O)CC1 c1(C(=O)NC2C(CNC(=O)C=C3CCOCC3)CC2)snc(O)c1Cl C1(OC)CN(Cc2nc(NS(=O)(=O)CC3CC3)cn2C)CCC1C(F)(F)F CS(=O)(=O)C(C(=O)N1CCC1CNC(c1cccc[n+]1[O-])=O)C1CC1 C(=O)(C(O)CCCNC(c1nnn(CC)c1C)=O)NC(c1noc(C)n1)CC c1(CC(N2C(C(C)(C)NC(CC=C)=O)CCC2)=O)c(Cl)cccc1Cl C(CC(O)CC(=O)N(C)CC1CCCN1C(C1CC1c1nnc(S)n1C)=O)SC N1(C(CN(C(C)=O)C)=O)CCC2(CCCN2c2ccc3nnnn3n2)C1 N1(C(C=C(CC)C)=O)CCC2(CCC(CNC(C3(C)CCC(=O)N3)=O)O2)CC1 C=CCCCCCCNC(=O)C(CC(C)C)ONC(=O)CC(C)OC.C(N)=O CC1(C2CC2)CN(C(=O)CN2CCCC2=O)CCO1.C12CCC(C1)NC2=O CCCC(CCC)=CC(=O)NC1CC(NC(=O)COC2CCCCC2)CC1O C(C(F)F)NC(C1(C(C)NC(=O)CC2CSC2)CC1)=O N1(C(c2c(C)csc2)=O)CCC2CN(C(=O)CNC(=O)CN(C)C)CCC12 C(=O)(C1=C(C)OCC1)N(C1C2CN(Cc3c(-c4cccn4C)cc[nH]c3=O)CC12)C N1(C(C2CCC(NC(c3cn(CSC4CC4)nn3)=O)C2)=O)CCC(C(C)=O)C1 C1(C(=O)NC2CCCCN(C(CCC(=O)NC)=O)C2)Cc2ccccc2S1(=O)=O S(=O)(=O)(c1cccc(S(=O)(=O)F)c1)N1CCCC2(N(C)CCC2)C1 C(c1cncnc1O)=CC(=O)N(CCC(C)NC(c1cncc(OC)n1)=O)C C(=O)(C1=Cc2ccccc2C1)N1CC(C)C(NC(C(F)=C(C)C)=O)C(C)C1 c1(C(=O)NCC2C3N(C(CC(C(C)C)C)=O)C(CC3)C2)cn(C)c(=O)nc1O N1(C(c2cc(C)c(C)o2)=O)CCCN(C(=O)C(F)C(F)(F)F)C(CC2CC2)C1 C1(NC(c2ccc(C(F)(F)F)nc2)=O)CN(C(=O)C=CCN2CCC2)CC1F N1(C(CN(CCOC)C(C2CCCCC2C)=O)=O)CCC(C)(CO)CC1 c1(C(N(C)CC2CCCCN2C2CCCC2)=O)cc(O)nc(=O)n1C c1(C(=O)NCCC(CCNC(CCOC)=O)C)c(F)c(F)c(F)c(F)c1F C1(C(N(C)CC2CCN(C(c3n(CC#C)ccc3)=O)CC2)=O)CC(C2CCC2)C1 c1(C(=O)NCC2CN(C(C=CC(C)O)=O)C2)ccc(S(C)=O)cc1 CCCCC(C(=O)NCC(F)CNC(c1ccccc1SC(F)F)=O)NC(N)=O CC1(C)CC(CC(=O)NC2CCOC2)CN1C(=O)CCC(F)(F)F C(CCC)(C(O)C(=O)N(C)C)CCCC(=O)NC(C(CC=CC)CC)=O N1(Cc2c(C)ccc(Br)c2)CCC2CC(C(=O)NCc3cc(Cl)ccc3Cl)C2C1 N1(C(CCCC(=O)OC)=O)CC2CCCC(CNC(=O)CC(F)(F)F)(C2)C1 C1(NC(C2CC(CCNC(c3oc(C)c(CO)c3)=O)C2)=O)CC(C)N(C)CC1C C#Cc1cncc(C(N2CCC(N(C(=O)C(C(F)(F)F)OC)C)C2)=O)c1 N1(C(C(C)OCCOC)=O)CC2(CC(NC(c3nc(Cl)sc3Cl)=O)CO2)C1 N1(C(CC(C)C(F)(F)F)=O)CCC2CCN(C(c3ccc(Cl)cc3)=O)C2C1 c1(NC(c2c(-c3cncc(CC)n3)c(F)ccc2)=O)cc([N+](=O)[O-])ccc1Cl O=C(C(O)C(CCO)c1ccccc1)Nc1ccccc1C1CCC1 CCC1=C(C(=O)NCC2(NC(=O)C(C)CSC(F)(F)F)CC2)CCCO1 C1(C(=O)NC(CO)CCC2CC2)(OC)CCN(C(c2cccc(O)n2)=O)C1 N1(C(c2cc(CCC)nc(O)c2)=O)CCC2(CCCN2C(c2ncoc2C)=O)C1 c1(C(=O)NC2(CNC(c3c(CC)[nH]cc3)=O)CC2)ccc(C(F)(F)F)cc1OC c1(C(N(C)CC2(O)CCCN(C(COC(C)=O)=O)C2)=O)nccc2[nH]ccc12 N1(C(CC2CC(NC(C(COC)OC)=O)C2(C)C)=O)CC2CC(C)(C)C2C1 C1(C)(CNC(=O)OC(C)(C)C)CCCN1C(=O)C1CC1.n1(CC(=O)N)cc(CO)nn1 Cn1c(C(=O)NC2(C)CC2)ccc1C1COCCN1C(c1ccns1)=O CCCCC(C(=O)N(CCCC(C)(F)F)C)NC(c1ccnc(OC)n1)=O C#CCCC(C(=O)NCC(C)OCC#C)NC(=O)C=C=C(C)C c1(CC)nc(C(=O)NC2CCN(C(c3ccccc3C(C)C)=O)C2)c(C)o1 c1(C(N2C(C)(C)C(CNC(C3CC3F)=O)CC2)=O)ccn2nncc2c1 C1(C(=O)NCC2CCC(NC(C3CCCCC3O)=O)C2)(COC)CCOCC1 C1(NC(CCCSC)=O)CN(C(c2cc(F)n[nH]2)=O)CCC1C CN1Cc2ccc(C(N3CCN(C(=O)COc4ccsn4)C4(CC4)C3)=O)cc2C1 N1(C(CC(CC)C)=O)CCC2(CC1)CCN(C(=O)COCP(C)(C)=O)CC2C c1(NC(=O)NC(c2ncc(C)[nH]2)C)cnn(C(F)F)c1C c1(C(=O)NCC23CCCN(C(COC)=O)C2CCC3)cc(Cl)c(Cl)c([N+](=O)[O-])c1 c1(OC)cc(C(=O)NCC(C)(C)NC(C2C3CCC(C3)C2C)=O)cc(Cl)c1O C#CCCCCC(=O)NCC1CC(CCn2cc(CC3(C)CC(F)(F)C3)nn2)C1 C1(C(C)=O)CC1(Cl)C(=O)NCC1CC1CC(=O)NCCC1CC1C C(=O)(CC(C)(C)C(=O)NC1CN(C(=O)C(C)C2=CCCC2)CC1C(F)F)OC c1(C(=O)NC(C(C)NC(C2CC(CC)(CC)C2)=O)C(C)C)cc2ccc(Cl)cc2s1 CC(C)CC(C)CC(=O)N1C2CCC1CN(C(C1CCc3ncnn3C1)=O)C2 CC1(C)C(=O)CC1C(N1CCC(CNC(=O)CSCc2ccncc2)C1)=O Cc1ccc2oc(C(=O)N(C3CC(NC(c4ccc(C(C)(C)C)o4)=O)C3)C)cc2n1 N1(C(C2(NC(C(CC(C)C)O)=O)CC(CO)C2)=O)CCOCC(C)(F)C1 N1(C(C2C(OC)CC2)=O)CCC2CCN(C(=O)C(C#N)C(C)(C)C)C2C1 c1(C(=O)NC2C(NC(C(C)Cc3ccc(C#N)cc3)=O)C2)ccnc2cc[nH]c12 N1(C(C2CN(C)C(=O)C2)=O)CCCCC(NC(c2ccc(C3CC3)o2)=O)C1 N1(C(C2CCCC(C)(C)C2)=O)CCC2CCN(C(=O)CCC(C)(C)[N+](=O)[O-])C2C1 c1(OCC(=O)NC2C(NC(CC3CC(OC)C3)=O)CCCC2)cc(F)cc(Cl)c1 c1(C(=O)NCC(CCOC)NC(C(C)OCC=C)=O)cc2ccccc2nn1 C1(CNC(CCN(CC)CC)=O)CCC(NC(=O)Cn2cc(C)cn2)C1 CC1CCN(C(c2cnn3c2CCC3)=O)CC1CNC(C1CC2CC2C1)=O CC1(C)CCN(C(=O)C2=CCCSC2)CC1CNC(C1CCOC(C(F)F)C1)=O C1(C(=O)NCC2(OC)CN(C(=O)CCS(C)=O)C2)Cc2cc(F)cc(F)c2O1 CCC(CC(=O)NCC(CC1CC1)OC)NC(=O)C(C)N=[N+]=[N-] c1(C(=O)NCC(CNC(C2C(C)(C)CO2)=O)F)ccc2cc(O)ccc2c1 N1(C(c2ccsc2)=O)CCn2nc(CNC(C34CCCC3CCC4)=O)cc2C1 C1(NC(CCC(=C)C)=O)CCC2CN(C(=O)C(C)=C3CCCC3)CCC2C1 CCC(C(=O)NCC1C=CC(NC(c2cccnn2)=O)C1)Sc1ccccc1 Cc1ccc(F)cc1CN1CCC(C(N2CCC(c3ccc(Br)cc3)CC2)=O)C1 c12nc3n(c1NC2=O)CCCC3.n1(CC)ncc2c1CCC(NC=O)C2 N1(C(c2cn(CCNC(C3ON=C(C)C3)=O)nn2)=O)CCc2cc(F)ccc21 C1(NC(C2(NC(C(CC3CC3)OC)=O)CC(F)(F)C2)=O)CCCC(O)CC1 c1(NC(=O)NC2CCc3nncn3C2)cc2c(cc1Br)CCNC2=O C1(OC)CN(C(=O)C=C(C)C2CC2)CC1NC(=O)CSc1cccc(F)c1 Cc1cccc(C)c1.Cc1nc(CNC(=O)N(C2CC2)CC2CC2C)cs1 C(=O)(C1=CCCCCC1)NC(C)C(C)(C)C(=O)NC(CN(C)C)CCO C1(CNC(CCc2ccnc(C)n2)=O)CC2(CCC2)CN1C(=O)CSC(C)C c12ccccc1S2.C(C(C)C(=O)NC1CC(CNC(C2CCCCC2)=O)C1)OC c1(C(=O)NCC2(C)CCN(C(C(CC3CC3)OC)=O)C2)nc2ccccn2c1F C1(CC(=O)NCC2CN(C(=O)CCOc3cccc(Cl)c3)C2)CCS(=O)(=O)CC1 CC(C(=O)N1CCN(CCC2(O)CN(C(=O)COCCOC)C2)CC1)C(C)(F)F N1(C(C(C)OCC#C)=O)CCC(CO)C(NC(c2cnnn2C)=O)C1 N1(C(Cc2n(C)nc(C(C)(C)C)c2)=O)C2CCC1CN(C(c1cc(F)cs1)=O)C2 Cc1cc(CCN=C(NCCn2ccnn2)NC2CCS(=O)(=O)C2)ccc1F c1(C(N2CCC(C)C(C(=O)OC)C2)C(=O)NC)cc(Cl)c2c(c1)OCCCO2 CN1CCC(NC(c2[nH]ncc2C#N)=O)C12CCCN(C(C1(F)CCOC1)=O)C2 N1(C(C(CNC(c2cccc(CC#N)c2)=O)N(C)C)=O)Cc2n[nH]cc2C1CO c1(CNC(C(CCOC)OC)=O)nc2c(s1)CCN(C(c1c(C)cnn1C)=O)C2 c1(CC(=O)N(CC(C)NC(C2CC(=O)N(OC)C2)=O)CC)csc2ccccc12 C(=O)(CCC(=O)NCCCC(C)(C)NC(C1CCCC1)=O)NCCC CCCCC(CC(F)F)NC(=O)OC(C)(C)C.N12Cc3[nH]nc(c3C1)C2=O c1(C(=O)NC2CN(C(C(CC)C(F)(F)F)=O)CC2(C)C)ccc2c(ccn2C)c1 C1(C(N(C2CC=CC2)C)=O)CCN(C(C2CCCC23CCC3)=O)CCO1 C(C(C)(C)C(=O)NCCCC(F)F)N(C(C(CNC(=O)OC)C)=O)C C12(C(=O)NCC(F)CO)CC(CO1)N(C(c1cnn[nH]1)=O)C2 Cc1oc(C#N)cc1C(N1CC(NC(C23CCC(C2)OC3C)=O)CC(C)C1)=O c1(CN(C(C(N2CCC(Cc3n(C)ncn3)C2)=O)=O)C2CC2)cccc(Cl)c1 C#CC(CNC(=O)C(c1cccs1)NC(=O)CCC1CCCCC1)CC C1(C#N)(C(N2CC(CNC(c3cc(C(C)C)c(F)cc3)=O)C2)=O)C(C#N)C1(C)C C(=O)(C1CCCc2nc[nH]c21)NC1C2CC3CN(c4c(C#N)cncn4)C1C3C2 Cc1c(NCCCN2CCOCC2=O)ncnc1NCCc1ccc(C(F)F)o1 CC(C)(C)C1=NOC(C)(C(N2CCC=C(CNC(C3CC3C(N)=O)=O)C2)=O)C1 N1(C(CCN(CCC)C)=O)CCC(C)(CC(=O)NCCC(O)COC)C1 C(CCCCCC(=O)N1CCc2sccc2C1)NC(C1CN(C(C)=O)C1)=O C(=O)(C(C#N)C(C)(C)C)NC1CCN(C(C=CCOC)=O)C1C Cc1ccc(C(=O)NC(CCN(C(=O)CCSC(F)(F)F)C)C(C)(C)C)cc1O c1(C(N(CC(CNC(C2(OC)CCC2)=O)C)C)=O)ccnn1CC(F)F N1(C(C2(C#N)CCC(=O)C2)=O)CCCC(O)(Cn2ccnn2)CC1 C1(NC(C(CC)OC)=O)CCCC12CCN(C(c1ccc(OC)c(F)c1)=O)CC2 C1(C(N(C(=O)CN2CCC(C(N)=O)CC2)CCSCC)=O)C(C)CCCNC1=O Cc1oc(C#N)cc1C(=O)NC1CC(NC(=O)CCOC2CCCCC2)C(O)C1 C12CC(C)N(C1)CS2.C1(CCC)CCCN(C(C)=O)C1 c1(CCCN2CCC(c3nc(C)on3)CC2)ccc(N(C)C)cc1C c1(C(C)(C)CNC(=O)CC#N)ccc2[nH]c(CN3CCC4(C3)CC4(F)F)cc2c1 c1(NC(CN(C(=O)NCC2CN3CCC2C3)CC)=O)ccc(F)cc1C Cc1ccc(CS(=O)(=O)NC(C)(C)CNC(=O)Nc2cnc(O)cc2C)c(C)n1 C1(N(C)C(c2ocnc2C(F)F)=O)CN(C(c2cn(C)[nH]c2=N)=O)CC12CC2 C=CCC(CC)C(=O)NCCCN(C(c1ccc(F)c(OCC(C)C)c1)=O)CC N1(C(C2C=C(C)CS2)=O)CCOC(C)C1C(N1CC(OCC(F)F)C1)=O C(=O)(C1CCCc2sccc21)NC12CC(NCc3nc(C)c(C)o3)(C1)C2 N1(C(c2c(C)nc3ccccn32)=O)CCCC(N=c2[nH]c(Cl)nc(C)c2Cl)CC1 C1(NC(c2nc(COC)sc2)=O)CN(C2CC2)CC1C.C12(CC1)C(=O)NC1(CC1)C2.CC N1(C(C(C)OCCC=C)=O)CC(O)CC1CC(=O)N(CC(C)(C)C)C1CC1 C(=O)(C(F)(F)C(O)C1CC1)NCC(C1CCCN1C(c1ccccc1)=O)(C)C N1(C(c2ccc(-c3ccco3)cc2)=O)CCc2cc(Br)ccc2C1 C1(NC(C(C)NC(N)=O)=O)CN(C(=O)C2=COCC2)CC2(CC2)C1 Cc1c(Cl)c(C(=O)NC2CCN(CCCNC(=O)C(O)C(C)(C)C)C2)nn1C c1(C(=O)NC2CCN(C(c3c(C)cc(=N)[nH]c3)=O)C2C)cn(C)c(=O)n(C)c1=O S(=O)(=O)(c1ccc(Nc2cc(F)ccc2F)nc1)N1C2(CCS(=O)(=O)CC2)CC1 c1(NC(C(c2cnn(C3CC3)c2)N(C(CC)C#N)CC)=O)ccccc1C C=CC(C)(C)CC(=O)N1CCOC(CC(=O)NCCC2CCCCCC2)C1 C1(C(N2C(C(C)C)CCC2)=O)N(C(=O)CC2(C)CCC2)CCC1(C)C N1(S(CCCC)(=O)=O)CCC(F)(F)C(C(=O)Nc2ccc(F)cc2C#N)C1 c1(C(=O)NCC2(NC(C34CC(F)(C3)C4)=O)CCOC2)cccc(CO)n1 C1(CNC(c2c(C)ncn2O)=O)CN(C(C2CC=CC2)=O)CC(C(F)(F)F)O1 C(N=c1[nH]c(=NCCC(=O)NC2CC2)[nH]c2c1CCCCC2)c1n(C)ncc1Cl C1(C#CC(=O)N(CC(=O)NCCC2CCCN(C)C2)C2CC2)(CC)COC1 CC1CC(C(=O)NC(C)C(C)F)N(C(=O)CCc2nncs2)C1 C12CCN(CC1)C(=O)C(=O)NC2.c1(OCC)cccc(OCCOC)c1 c1(OC)ccc(CS(=O)(=O)NC(C)CS(=O)(=O)N(C)C)cc1Br N1(C(c2n(C)c(O)nc2)=O)CCCC12CCC(NC(C1(S(C)(=O)=O)CC1)=O)CC2 c1(NCc2c(C(=O)OC)oc(C)n2)ccc(CSC2CC2)cc1[N+](=O)[O-] CC12CC(C(=O)NCc3ccc([Si](C)(C)C)cc3)(C1)C1(CCOCC1)O2 C1(CNC(c2cn(CC)nn2)=O)CN(C)CCN1C(=O)CCc1ccccc1F CCCC(C(=O)NOCCCC(F)(F)F)NC(c1cnn(C(C)C)n1)=O C1(NC(COCC(=C)C)=O)CCCC12CN(C(=O)C(c1ccc(C)cc1)C)C2 O=C(CCN=C(NC1CC2(CC2)C1)N1CCC2(CCOC2)C1)N1CCCC1 C1(NC(=O)C(F)C2CCC2)CC2(C1)CC2C(N)=O.C12(CCCC1)CCC(=O)N2 C(C)(C(C)C(=O)NC1(CO)CC1)NC(CCCOCC=C)=O c1(C(N2CCC(CNC(CCC(C)OC)=O)CC2C)=O)c[nH]c2cc(Cl)ccc12 C1(NC(CC(CNC(=O)Cc2cccnc2C)OC)=O)CC2CC1OC(=O)N2 CCC(CC(=O)N1CCCC1C(C)NC(=O)CSC(C)(C)C)CC(C)C C12(NC(C3ON=C(C)C3)=O)CN(C(=O)C=Cc3ccncc3)CC1CS(=O)(=O)C2 c1(CC(=O)NC2CN(C(C3(C#C)CC3)=O)C2)cccc(F)c1 C(=O)(CCC(C)(F)F)NC(C)C(=O)NC(CN1CCCC1)CO CC1CCCc2cc(C(=O)NCC(O)CNC(C34CCCCC(F)(C3)C4)=O)nn21 C12(NC(COCCC(C)C)=O)CCC(CN(C(c3cc(Cl)ccn3)=O)C1)C2 c1(OCC(=O)NC(CCCNC(C(C)C#N)=O)C)ccc(CO)cc1 CC1(C)CN(C(=O)CCF)CC2(CN(C(c3ccc(=N)[nH]c3Cl)=O)C2)O1 c1(CC(=O)NC2CCCC(CNC(CN(CCC)C)=O)C2)ncn2c1CCC2 N1(C(c2n(CC)cnn2)=O)CC2(COC(CNC(c3ccc(C)c(Cl)c3)=O)C2)C1 C1(CCC)CN(C(c2c(C)cccc2F)=O)CCN1C(=O)COc1cccnc1 Cc1cc(N(C)CCOC(C)(C)C)nc(=NCCc2csc(Br)n2)[nH]1 c1(CC(=O)N(CC(CC)NC(=O)Cc2ccn(C)n2)C)cnn(C(C)C)c1 C1(C(=O)NCCN(C(=O)CN(S(C)(=O)=O)C)CC)CC(C(C)(C)C)=NO1 N1(C(C(CC)(C)O)=O)CCCC(N(C(=O)C(=Cc2c[nH]cn2)F)C)CC1 N12CC(C)OC3(CCN(C3)C(=O)CCCCC1=O)C2.CC(=O)N(C)C(C)C C1(C)(C(N2CCC(C(=O)OCC)C2)=O)CN(C(=O)CSC(F)(F)F)C(C)(C)C1 C1(C(N2CCC(C3CCCN3C(C3CC4(CC4)C3)=O)C2)=O)CCOCC1 c1(CCC(=O)NC(CN(C(C(C2CCCC2)OCC)=O)CC)C)ccnc(C)n1 c1(C(N(CCC(C)NC(=O)C(C)(F)C(C)(C)F)C)=O)cn2ncccc2n1 c1(C(N2CC(C(=O)NCCc3ccc(CO)cc3)C2)=O)cccc(=O)n1O N1(C(c2c(C)ccs2)=O)CCC2(CC(NC(C3CC34CC(F)(F)C4)=O)C2)C1 c1(NC(c2cn(CCCC)nn2)=O)ccc(Cc2ccccc2)cc1 C1(C(N)NC(=O)COCC2CC2)CCCCO1 C(=O)(CNC(=O)CC1(CSCC2CC2)CC1)N(C)CC1C(CC)C1 N12CCN(CC1)CCC1(CC1)C2=O.c1(C(C(=O)NC)=O)cscc1Br Cc1cc(Cl)c(C(N2CC(NC(=O)CSCc3ccc(Cl)cc3Cl)C2)=O)cn1 c1(CN(C(c2cnc(CC)s2)C(=O)NCC=C)C)cccc2c1OCO2 CCC(CC)(CCNC(=O)CS(=O)(=O)NC1CC1)NC(c1[nH]ccc1C)=O CC1CN(C(C23COCC2C3)=O)CCN1C(=O)Cc1ccc(O)cc1Cl c1(CC(=O)NC(CC)CN(C)C(c2cscc2Cl)=O)ccnnc1O C1(CC(=O)NCC2N(C(C3N(C)CCCC3)=O)CC(O)C2)CCC(C)(C)CO1 Cc1cc(C)c(C#N)c(N2CC(NC(C3CCN3C(C)(C)C)=O)CC(C)(C)C2)n1 C1(C(=O)NCC2CCCCN(c3c(C)c(Cl)ncn3)C2)CCc2nnnn2C1 C1(NC(CCOC)=O)CC(NC(c2c[nH]c(C(F)(F)F)c2)=O)C12CCC2 N1(CCNC(C2C(COC)C2)=O)CCCN(C(=O)C(F)CC2CCOC2)CC1 C1(O)(C(C)NC(c2cc(CCCO)on2)=O)CCN(C(C2CCC(C)O2)=O)CC1 C1(C(N(C(C(=O)OC)(C)C2CC2)C)=O)CN(C(=O)COCCOC)CC(C)O1 c1(C(N2CCC3C(NC(CC4C(C)=NN(C)C4=O)=O)C32)=O)n[nH]c2cccnc12 c12cc(nc(CO)n1)N2.N1(C(c2cnccn2)C)CCN(CC2CC2(C)C)CC1 c1(C(=O)NC2CC(C)N(C(=O)C=CCF)CC2)cc2c(cc1Cl)OCO2 c1(SC(C)(C)CNC(=O)NCc2ccccc2)ccncc1 C1(F)(CNC(C2(C(=O)NC)CCC2)=O)CC(NC(=O)CC2C=CCC2)C1 C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC2CCC1N2C(c1csc2c1CCCC2)=O Cc1nc2ccc(C(N3CCC(CF)(NC(=O)C(C)NS(C)(=O)=O)C3)=O)cn2n1 N1(C(=O)NCCOC)CCN(C(c2cn(C3COC3)nn2)=O)CC1CC(F)F C(=O)(C#CC1CC1)NCCCN(C(=O)CC(c1ccc(OC)cc1)C)CC C#Cc1ccc(Cl)c(C(=O)NCC(O)CNC(=O)C(F)C2CCCC2)c1 C(=O)(C(C)(C)CC(C)C)NCC1CCCC(NC(c2cccc(NCC)c2)=O)C1 CC1(CNC(=O)CCc2ccccc2N)CC(F)(F)CN1C(=O)C=CC1CCC1 C1(C(=O)NCC2(C)C(C)CN(C(=O)Cn3ccnn3)C2)CCCN2CCCCC12 c1(C2(C(N(CCc3cn(C(C)C(=O)O)nn3)C)=O)CC(O)C2)ccccc1F Cc1cc(F)c(NC(C2CC2NC(=O)Cc2ccc(F)cc2)=O)cc1F c1(C)noc2c1CC(C)CC2.C(C(=O)OC)N(C(=O)CNC(=O)NCC1CC1)CC#C c1(CC)cnc(C(N2CCN(CC3CC(OC)C3)CC2)C(=O)NCCC#N)nc1 CC1CC2(CCN(C(=O)CC(Cl)Cl)CC2)CN1C(=O)CCC1CCC(=O)C1 N1(C(c2c(OC)scc2)=O)CCC(CNC(=O)C(C(C)(C)C)NC(C)=O)C1(C)C C1(CNC(CCN(C(COC(CC)(C)C)=O)CCCO)=O)(CO)CC=CC1 C12CCCC(CC1)NC2=O.c1(CN)cc(C2CC2)no1.C(C(=O)N)N(C)C(N)=O c1(C(=O)NC2CCC(NC(C3C(C)=C3)=O)C2)ccc2n[nH]c(C)c2c1 c12ccc(I)c(c1)CCC(=O)N2.C1(CC)CCN(CC2CCCN2C(C)C)CC1 c1(C(=O)NC(C2CN(C(=O)COC3CCOC3)C2)C)cnc2ccccc2n1 C1(NC(c2ccn3c2CSCC3)=O)CC2CC(C1)N(C(C1CC1(F)F)=O)C2 n1(CC)cc(Cl)c(C(N2CCC(Cn3cc(CN(C)C(C)=O)nn3)C2)=O)n1 C1(NC(c2ncn(CC)c2)=O)CC2CC(C1)N(C(=O)C(C)(F)c1ccccc1)C2 N1(C(C2C(C)(C)C2)=O)CCC(NC(=O)CCC2CCCCC2)C(C(N)=O)C1 c1(CC)oc(C(=O)NC2CC(C)N(C(c3cn(CCO)nn3)=O)C2)cc1C Cc1cc[nH]c(=N)c1C(N1CCN(C)C(CNC(C2(Cl)CC2(F)F)=O)C1)=O N1(C(C2N(C(C)=O)CCC2)=O)CC(NC(C2CC2(F)F)=O)C(F)(F)C1 C(c1sccc1Br)=CC(N1C(CNC(C2CCN(CC)C2)=O)CC1)=O CC1(NC(=O)CSC2CCCO2)CCCN(C(=O)Cc2ccc(Cl)cc2)C1 N1(C(C(C)NC(CC)=O)=O)CCCCC(N(C)C(c2ccncc2N(C)C)=O)C1 CC1CC(=O)CC(C(=O)O)N1Cc1cccc(C(F)(F)F)c1Cl c1(C(=O)NC(C(C)(C)C)CO)cnc2c(C3=CCCCC3)cnn2c1 C1(C(=O)NCC2(C(=O)NCc3cc(CO)on3)CC2)COCCOC1 CC1CC=CCC1C(=O)NCc1cccc(C(=O)NOCC2CCCC2)n1 Cc1ccc(-c2csc(NC(=O)CSC3CCC(=O)N3C3CC3)n2)cc1 c1(C(N2CC(NC(C3(CC#C)CC3)=O)C3C2C3)=O)ccc(S(N)(=O)=O)cc1F N1(CC(=O)NC(C)C)CCCC(NC(C2CCCS2)=O)CC1 Cc1ccc(C(N2CC3C(CNC(=O)C(C)Oc4ccccc4)C3C2)=O)c(N)n1 c1(NC(c2n[nH]c3c2CN(C(C(C)S)=O)C3)=O)nc2ccc(C(F)(F)F)cc2o1 c1(C(=O)NC2C(CNC(CN(C(=O)OC)C)=O)C2)cn(C)[nH]c1=N N1(C(CN(C)CCO)=O)CC2CCC1C(CNC(C1(C)CC(O)CN1C)=O)C2 c1(CC(N2CC(C)(CC(=O)NCC3CN(C)C3)C2)=O)ccc(F)cc1 c1(NC(C2N(C(CC(=O)OC)=O)C3C(C2)C3)=O)ccc2cnoc2c1 N1(C(c2cn(CC)nc2)=O)CCC(C(C)CNC(C2CC(=O)C2C)=O)CC1 CC1CCN(C(c2cc(F)ccc2Br)=O)CCN1C(c1cnn2c1CCC2)=O Cc1ccc(F)c(C(=O)NCC2CC2NC(c2c(C)ncn2C)=O)c1 CC1(C(N2CCOC3(C2)CN(C(C2CC(F)C2)=O)C3)=O)C2Cc3ccccc3C12 c1(OC)ccc(S(=O)(=O)NC2CC(CNN3CCCS3(=O)=O)C2)c2ccccc12 NS(=O)(=O)CCCCCCCCCNc1cc(C2CC2)cc(F)c1 CCCC(C)CC(=O)N1CC(CNC(c2cn(C3CC3)cn2)=O)C(C)(C)C1 c1(NC(C2C(C)(NC(C(C(C)(C)C)NC(C)=O)=O)CCC2)=O)cc(C)cc(C)c1O C12(C(=O)NC(C(C)NC(C3CCC3c3nc(S)n[nH]3)=O)C)CCC(=O)N1CCS2 CC1C(C(=O)NCC2CN(C(c3cnn(CC4CC4)c3)=O)C2)C(O)C(=O)N1C c1(NC(c2nc(CCC)oc2)=O)ccc(CC)c(OCCSC)c1 c1(N(C)CC2CCCN(C(C=NOC)=O)C2)nn2cc(C)nc2s1 C(=O)(CCCN(C)N=O)NC1CCN(CCNC(C(C)(C)OC)=O)CC1 N1(C(C2CC(C)(CC)C2)=O)CCOC(CCCNC(c2cnc(C)[nH]2)=O)C1 CC1(C)CCCOC1C(N1CC(OCCC(N2CC3(CC3)CC2CO)=O)C1)=O c1(COC)nccc(N2CCCC(C(=O)NC(CC)C(C)C)C2)n1 n1(CC)nc(C(C)C)cc1C(=O)NC1CCC1CNC(=O)CC(C)OC c1(C(N(C(C)CNC(=O)CCC2CCN(C)C2)C)=O)cn(C)c2ccccc12 CN1CC(NC(c2ccoc2CNC(c2ccns2)=O)=O)CC1=O N1(C(C(C)OCC#C)=O)CCN(C(=O)C=Cc2cncs2)C(c2ccncc2)C1 N1(C(C(C)SC(F)(F)F)=O)CCC(O)(CCNC(c2ccsc2Cl)=O)C1 c1(C(=O)NCCCN(C(C(CC(C)C)NC(C)=O)=O)C)cnc2ccccc2c1 C1(NC(CN(CCSC)CC)=O)CCN2CCCCC12 c1(C(=O)OC)cc(C(=O)N(CC(C)(C)CNC(=O)C(O)C2CCC2)C)c(F)cn1 C(C)(CNC(=O)C(C)CC#N)(CC(C)C)NC(c1cc(CC)nn1C)=O c1(OC)cc(F)c(C(N2CC(CNC(c3ccco3)=O)C3CC23)=O)cc1OC C1(O)(CN(C)C(c2cscc2Cl)=O)CCN(C(C2CSC2)=O)CC1 CC1(C)CC(C(=O)NC2CC3(CC3)C2)CN(C(=O)C(C)(C)CCF)C1 C1(C(C)C)CN(C(=O)OC(C)(C)C)CCN1Cc1ccccc1-c1nn[nH]n1 N1(C(C(C(=C)C)(C)C)=O)CC2(CC(NC(c3cccc(F)c3SC)=O)CO2)C1 c1(CC)ccnc(C(N2CCN(C(=O)CNC(c3ncc[nH]c3=O)=O)CC2)=O)c1 C1(C(=O)NC2CC(O)C(O)C2)(COC)CCN(C(c2ncccc2F)=O)C1 C(C(=O)NC(CCN(C(=O)CCCn1cncn1)C)C(C)C)(C(C)C)OCC C1(C(=O)NCCC2(OC)CN(C(C=C(CCC)C)=O)C2)CC12CCCC2 Cc1[nH]nc(Cl)c1C(N1CCC(C2CCCN2C(c2ccncc2)=O)CC1)=O N(C1CCCc2cc(C(C)(C)C)ccc21)C(C)C C1(CC(=O)N(CCCC)CC(C)C)C2CN(C(c3nc(CC)oc3C)=O)CC12 C1(C#N)(C(=O)NC2CN(C(CC3ON=C(CC)C3)=O)C2)CC2(CCC2)C1 Cc1nc(C2CC2)nc(O)c1C(=O)NC1CCC1NC(=O)C=CC1CCCN1C c1(C(N(CC(=O)N(C(C)CC2CC2)C)C2CCC2)=O)cnccn1 C1(CC)C(NC(c2cc(SC)c(C)o2)=O)CCN1C(=O)Cc1csc(S)n1 CP(C)(=O)COCC(=O)NCCCCCNC(=O)C(N1CCCCC1)C1CC1 C1(C(=O)NCC(CC)OC)CC2(CC(NC(=O)C(C)Cc3ccc(F)cc3)C2)C1 N1(C(C(C)OCCC=C)=O)CCC(F)CC1C(=O)NCCCF c1(OC)cnc(F)c(C(N2CC3CC3(CNC(=O)CNC(=O)C3CC3)C2)=O)c1 CC1(C)CC(NC(C2CCCC3(CCC3)C2)=O)CCN(C(=O)Cc2ccsn2)C1 CS(=O)(=NC(=O)c1cc2c(cc1Cl)NC(=O)CO2)c1ccccn1 C(C)(CCC(=O)N1CSCC1C(=O)N(CCCC(O)CO)CC)OC CC(C(=O)NC(C)(C)CCNC(C1CC(=C2CC2)C1)=O)C(C)n1cccn1 CCCC(C)CC(=O)NC12CCCC(NC(=O)CC(CC)SC)(C1)C2 CC1CCCCN1C(c1ccc(NC2CC2C(=O)NCC(N)=O)cc1)=O n1(CC)cnc(C(=O)NC(CC2CC2)C(=O)NCc2nc(C(C)C)n[nH]2)c1 c1(C(C(=O)NC(CN(C(=O)Cc2ccno2)CC)C)(F)F)ccc(Cl)cc1Cl c1(C(=O)NC2CN(Cc3ccsc3)CC2F)cc(Cl)cc([N+](=O)[O-])c1Cl C1(C(N2CC(CN(C(=O)CCC3CCCCO3)C)C2)=O)CCn2c(O)nnc2C1 c1(CS(CC(C)C)(=O)=O)n[nH]c2c1CN(C(=O)NC13C=CC(CC1)C3)C2 C(C(=O)NC1CN(C(=O)CC(C)(C)C)CC1C(F)F)(C(C)(C)C)OC c1(CC(N2C(CCCNC(CCOC)=O)CCC2)=O)noc2ccccc12 C1(NC(c2c(S(C)=O)cccc2)=O)CCN(C(C2(C(N)=O)CC2)=O)CC12CCC2 C1(OCCNC(C2(CC)CC2)=O)CCN(C(C2(c3ncccc3F)CC2)=O)CC1 c1(CNC(COC)=O)c(C)nn2c1CN(C(=O)CC1CC3(CC3)C1)CC2 C=CC1CN(C(=O)OC(C)(C)C)CC1C(N1CCCC1c1cncnc1)=O N1(C(CC=C=C)=O)CCC(NC(c2cc(Cl)ccc2C)=O)C(CO)CC1 CCC(CC)C(C(=O)NCC1(NC(=O)CCC(C)OC)CCOCC1)OC N1(C(c2cccc(C(C)(C)C)n2)=O)CCC(NC(=O)C=Cc2cc[nH]n2)C1(C)C c1(NCC2CCC(NC(C(C3CCOC3)OC)=O)CC2)ncc(C)c(SC)n1 Cc1ccc(NC(=O)CC2(C)CCN2C(=O)CC2COCC2O)cc1O CC1(C)CC(CNC(=O)Cc2ccoc2)N(C(C2(C#N)CCC2)=O)C1 C12(C(=O)Nc3c(C(C)C)n(C)nc3)CCC(NC(C3CN(C)CCO3)=O)(CC1)CC2 CC1CN2CCN1CC2C(=O)NC1(CNC(c2cnccc2C(F)F)=O)CC1 C1(NC(C(C)NC(C(C2CCC2)OC(C)=O)=O)=O)C2CCC(F)(F)C12 N#Cc1cccc2cc(-c3cccc4[nH]c(C(=O)NCCNC=O)cc34)cnc12 c1(C(=O)NC2C(NC(=O)Cc3cnccn3)C2)ccc(F)c(CO)c1 O=C1CCN(CC2CCOC2)C(=O)N1NC(c1cc(C(c2ccccc2)O)on1)=O c1(C(=O)NC2CN(C(Cc3cnc(C)s3)=O)C2)ccn2ncc(C)c2n1 CCCC(O)CC(=O)NC(C)CC(C)NC(=O)CN1CCc2ccccc21 c1(C(N(CC(=O)N(CCN=[N+]=[N-])CC)C)=O)c(Cl)cnn1C C1(NC(C2C(C#N)C2)=O)CCCN(CC(=O)NCCNC(N)=O)C1 C(=O)(C1=CC(C)(C)C1)NCC(CC1CN(C(C(C)OCC2CCOCC2)=O)C1)(C)C N1(C(CC=C=C)=O)CC(C)(C)CC1CC(=O)NCc1nc(C)c(CC)o1.C(N)=O C(CS(=O)(=O)CC(=O)NCC1CC(O)(C(=O)NC2CC3(C2)CC(O)C3)C1)OC c1(NC2CC3OC(=O)OC3C2)cccc(S(F)(F)(F)(F)F)c1 c1(C(C(N2CC(C(C)(C)O)OCC2)=O)=O)ccc2c(c1)CCC2 c1(NC(C2N(S(c3cn(CC)nc3)(=O)=O)CC(C)C2)=O)cc(C)c(Br)c(F)c1 c1(CC)ccc(C(N2CCC(C)(NC(c3ocnc3CC)=O)C2)=O)cc1F C1(NC(C(C)C(F)F)=O)CN(C(=O)C=C2CCSCC2)CC(F)(F)C1 c1(C(N(CC(C)NC(C2CCNC2)=O)C)=O)cnc2c(c1)CS(=O)(=O)CC2 c1(CCC)cc(C(=O)N(CC(O)CNC(=O)CNC(=O)CC)C)n[nH]1 N1(C(CN(C(=O)OCC)C)=O)CC2CC1C2C(N1CC(N2CCNC2=O)C1)=O c1(CC)nn(C)cc1C(=O)NC1CCN(C(=O)CC2CCC(=O)CC2)C1C C1(C(=O)OC(C)(C)C)(CO)CCCCC1.N1(C(C)C(=O)N2CCC2CN)CCCCCC1 C1(NC(C(=O)NC(C)C)=O)CC(NC(=O)CC2(C#N)CCCCC2)C12CCC2 C1(C(N2C(C3(O)CN(C(CC(C)OC)=O)C3)CCC2)=O)CC(=O)N(C)C1 c1(C(=O)NCC2CN(C(c3c(CC)noc3)=O)CC2C)cc(C#N)c(F)cc1F C12C(C1(C)C)C(=O)NC(C)(C1CC1)CNC2=O.C(CC(=O)OCCOC)=CC N1(C(Cn2ncc(C#N)c2)=O)CCC2CN(C(c3ccoc3Cl)=O)CC2C1 CCC(C)CCC(=O)N1CC2CC1CN2C(c1c[nH]cc1C(=O)OCC)=O c1(OC)ccccc1CC(COC)C(C)C.n1(CC(=O)O)cccnc1=O Cn1ccc2cc(C(N3CC4CCC(Nc5nnccc5C#N)C4C3)=O)cnc12 Cn1cnc2ncnc(NC3CC3CC(=O)O)c12 C(=O)(C(C)(C)C(F)F)N(C(C)CCNC(c1ccncc1Cl)=O)C N1(C(c2n(CCCC)ncc2)=O)CC(C(F)(F)F)C(CNC(=O)COCCC)C1 N1(C(c2cc(C)sc2C)=O)CCC(O)(CN(C)C(C2(C#N)CCCO2)=O)CC1 C(=O)(CCCCCF)NC1CC(O)(CNC(Cc2ccc(NC(C)=O)cc2)=O)C1 Cc1ccc(CC(=O)NC2(CNC(C3C=CC=CC=C3)=O)CCOCC2)c(Cl)c1 N1(CCC(=O)N(C)CCOCCN(C)C(C2CSCCS2)=O)CCCC1=O N1(C(C2C(=C)C2)=O)CCC(CNC(=O)CC2=CCCCC2)C(F)(F)CC1 N1(C(c2c(C)coc2)=O)CC(CNC(C23CCCN2CCC3)=O)CC1(C)C c1(CC)ccccc1C(=O)NCC1(O)CCN(C(=O)CCCc2cnccn2)C1 c1(C(N2C(C)CC(NC(c3cnc(S)nc3)=O)CC2)=O)cc([N+](=O)[O-])nn1C c1(CN2CC(C)(C)OC3(C2)CNC3)ccc2c(c1)CCC(=O)N2 c1(C(C(=O)NC2CCN(C(C(CCSC)O)=O)C2)(C)C)ccc(F)c(F)c1 C1(CNC(C(C)OCC2CC2)=O)CCCCC1NC(=O)C(F)(F)c1cnn(C)c1 c1(C(=O)NC2(C)CN(C(c3ccoc3C3CC3)=O)C2)ccccc1C(F)F N1(C(c2cncc(C#N)c2)=O)CCC2(CCC2)C(NC(c2ccc(CO)cc2)=O)C1 C1(C)(CC(=O)N(CCN(C(CC=CCC2(NC(C)=O)CC2)=O)C)C)CCCCC1 Cc1[nH]nc(Cl)c1C(=O)N(C(C)CNC(c1ncccc1C(C)(C)C)=O)C N1(C(CN2C(C)CC2)=O)CCC(CCNC(=O)CCc2ccc(Cl)s2)C1 c12cc[nH]c1C(=O)NC2.c1(C(CO)NC(CCNC(C)=O)=O)cccnc1 CC(C)CC(C)(CNC(=O)CC1CC=CC1)NC(C1CC2CCC1O2)=O c1(C(N2CC(C)C(NC(=O)CC3CCC3(C)C)C2)=O)cnn2c1C(=O)NCC2 Cc1cc(C(N2CC(O)(CCNC(=O)C(C)Oc3ccccc3)C2)=O)cc(C)n1 C#Cc1cc(C(=O)NC(CNC(=O)Cn2cnnc2O)(CC)CC)cc(N)c1 CCC(CC)CC(=O)NC1CN(C(=O)C(C)SC(F)(F)F)CCC1C(F)(F)F c1(NC(=O)CC(CC2CC2)NC(c2csc(O)n2)=O)cnc(O)c(F)c1 c1(NC(C)=O)ccc(C(=O)NC2CCC2NC(=O)CC2CC3CC3C2)cc1F N1(C(CCc2c(C)cccn2)=O)CCC2(CC(C(=O)N3CC(F)C(F)C3)=NO2)C1 C1(CCOC)CC(N=c2cccc(S(=O)(=O)NC3CC4CCC3N4C)[nH]2)CCO1 c1(C(N(CCCN(C(=O)COCc2ccsc2)C)C)=O)cccc(Br)c1 C1(C#CC(=O)NC2(CO)CCCN(C(C3(O)CCSC3)=O)C2)(CC)COC1 CCC(C)C(C(=O)NC(C(=O)NCCCCC(C)(F)F)C(C)C)N(C)C C(Cc1cnc[nH]1)(C(=O)NCC1(C)CCCO1)NC(C(C)=C(CC)C)=O N1(C(c2ncc(C(F)F)s2)=O)CCOC(C(N2CCOCC2)=O)C1 N1(C(C2CN(C)C(=O)N2)=O)CC2OCC(NC(=O)CCCc3cccs3)C2C1 C1(C(=O)NCC2CCC(CO)CC2)CC2CCC1N2C(c1c(F)cncc1F)=O N1(C(c2c(C)cncc2)=O)CCN(C(C2CCC(F)(F)CC2)=O)C(C)CC1C C(=O)(C(F)CCC(C)(C)C)N1CCC(C(N(C)Cc2onc(C)n2)=O)CC1 c1(C(=O)NCC23CC(NC(C4CCCOC4)=O)(C2)C3)cc2cccnn2c1 N1(CCCC)CCCCC1C(=O)NCC(C)N(C(=O)CC(C)F)CC c1(NCc2ccc(COCC)cc2)nc(N2CCCC(F)CC2)nc2sccc12 N1(Cc2ccc(OC)cc2F)C2CCCC1CN(C(=O)C(C)c1ccsc1)C2 N1(C(CCSC)=O)CCN(C(c2nc(O)sc2C)=O)C(c2cccc(Cl)c2)C1 c1(Cc2nc(C)on2)ncccc1NC(=O)C(=O)NC(c1ccn(C)n1)(C)C CC1=C(C(=O)N(C)CCOCCN(C)C(c2c[nH]c(=N)nc2C)=O)CCCC1 C1(C(N(C2C(OC)COC2)C)=O)C2CN(C(=O)CCc3nccs3)CC12 N1(C(c2ccnc(C(C)C)n2)=O)CCN(C(c2ncccc2Br)=O)C2CC12 C1(CC#C)(C(N2CC(F)C(F)C2)=O)CCN(C(c2cscn2)=O)C1 N1(C(c2c(C)cc(F)s2)=O)CCCC(NC(C2(CCF)CC2)=O)CC1 CCC(CC)(CC)C(=O)N1CCC(O)(C(C)NC(c2c(C)cc(=O)oc2C)=O)C1 n1(CC(C)N)cc(NC(=O)CC2CCCS2)cn1 c1(C(=O)OCC)cnc[nH]c1=NCC1CC(C)(C)CCC1NC(=O)C(O)C1CC1 C1(CNC(C2CCC2)=O)CC(F)(F)CN1C(C12CCCC(C1)OC2)=O CC1(C(=O)Nc2cccc(NC(=O)Cc3ncc(F)cc3F)c2)CCCC1(F)F C1(C(N2CCCC(=C)C2)=O)CCN(C(C2CC3CCC3C2)=O)CC1O C(=O)(C1=CCS(=O)(=O)C1)NC1C(NC(c2cnc(=N)[nH]c2)=O)CCCC1 CC(C(C)C(=O)N1CC2(C1)SCCC2NC(=O)CC(=O)N(C)C)S(C)(=O)=O c1(CC)nc(C)ncc1C(=O)NC1CC2CC1N(C(c1cn(CC)nn1)=O)C2 c1(-n2c(C(=O)NCC3C(NC(C4C(Cl)(C(=O)OC)C4)=O)C3)cnc2)ccccc1C N1(C(C(CN(C(C)(C)C)C)NC(=O)C2CC2)=O)CC(C)C1(C)C N1(C(Cc2ncc(C)s2)=O)CCOC(C(C)NC(C2CC(C#N)C2)=O)C1 c1(C(CSC)NC(=O)CNC2(C)C=CCC2)ccc(C)cc1 C(=O)(CC1=NN(C)C(=O)C1)NCC(N(C(COCCCCC)=O)C)C1CC1 C(c1cc(F)c(F)c(F)c1)=CCC(=O)NOCC(=O)NC1(C(=O)O)CCC1 Cc1ncc(NC(=O)CC2CCCCN2C(C2C(C)(C)C2(F)F)=O)c(C)c1C C1(NC(C2(CCC)CC2)=O)CCCCCC1NC(=O)Cc1ncn(C)c1C c1(N2C(CC(=O)OC)CCCC2)ncnc(NC2CCC(C)(C)C2)c1C Nc1cc(C(N2CCCC(F)(CNC(=O)C(O)Cc3cnc[nH]3)C2)=O)ccc1Cl C=CCCN=C(NCC(O)CN1CCC(C)CC1)NC1CC1c1cccc(C)c1 C1(NC(c2c(CC)snn2)=O)CN(C(=O)Cc2ccc(F)cc2)C(C)(COC)C1 N1(C(C23N(C(c4c(OC)nsc4)=O)CCC2CCC3)=O)CCn2cnnc2C1C C1(Nc2nnc(C)s2)CCN(C(=O)CCc2c(C)noc2Cl)C(C)C1 Cc1nn2cccnc2c1C(N1CCC(C)(CNC(=O)C(F)=CC2CC2)C1)=O c1(C(=O)NC(CNC(Cc2ccc(OC)cn2)=O)C2CC2)c(F)ccc(F)c1Cl Cc1c(Cl)ccnc1C(=O)NCCCN1CCN(C(=O)Cc2cn[nH]c2)CC1 C1(COC)CN(C(c2ccnn2C)=O)CCN1C(=O)Cc1cnn(C(C)C)c1 C=CCC(C(=O)N1CCCCC1c1n[nH]cc1C(=O)NC1(C)CSC1)C(C)C CON1CCC(C(N2CCC2C2(NC(c3cc(Br)n(C)n3)=O)CC2)=O)CC1 c1(CCC)cc(C(N2CC(C(N)=O)(CNC(=O)Cc3cnoc3)C2)=O)ccn1 c1(C(N2CCCC(CNC(c3cc(CN(C)C)on3)=O)C2)=O)nccc(Cl)c1O c1(C(=O)NCC2(C)CCC(NC(CCOCCC)=O)C2)cccc2[nH]c(=N)oc12 CC1(C)CCc2oc(C(NC3=COCCC3)=O)cc2C1C C12(NC(=O)NCCCC3(COC)CC3)CCN(C)CC1CN2C(=O)OC(C)(C)C CCCCCS(=O)(=O)CC(=O)N1CCCC1CN(C(=O)CN(C)CC)C1CC1 CC1(NC(=O)Cn2ncc(Br)n2)CCN(C(C2CCC(=O)N2)=O)CC1 c1(CC)cc(F)ccc1C(=O)NC(CCN(C(=O)C(C1CC1)OC)C)C(C)C c1(C(=O)NC2CCN(C(CCN(CCC)C)=O)C2)c(C)cc(C#N)cc1C c1(CNC(C2OCCN(C(c3scc(C)n3)=O)C2)=O)cnc(F)cc1C Cc1cccc(NC(C2CC3CC3N2C(c2cc[n+]([O-])cc2)=O)=O)n1 CC1(C)CN(C(c2cc3n(n2)CCC3)=O)CCC1NC(=O)C=CI c1(NC(C2(CNC(c3cccc(F)c3)=O)CC2)=O)cc(C(F)(F)F)ccc1CO c1(OC)ccc(C2CC(O)CN2S(=O)(=O)CCCOc2cccc(C)c2)cc1 Cc1c(C(N2CC(C)(NC(C3CCC=CO3)=O)C2)=O)cncc1Cl c1(C(=O)NC2C(NC(Cc3nc(COC)sc3)=O)CCC2)ccc2cnnn2c1 c1(CC)cc(Cl)ccc1NC(C1(CC2(CNC(C3CC3(F)CC)=O)CC2)CCC1)=O c1(C(=O)NC2C(C(N(CCS(C)(=O)=O)CC)=O)C2)c(Cl)cc(Cl)cc1Cl c1(CC)cc(C(=O)NC2CC(C(F)C(=O)NC(C)COC)C2)ccn1 C1(CC)C(NC(=O)CCC#N)CCCN1C(=O)C(C)n1cncn1 c1(NC)cnncc1C(=O)Nc1cnn(C)c1-n1cccc1.C1C(=O)N1C1CC1 C1(CC(=O)OC)CN(C(c2cnnn2CC)C(=O)NC2CC2)CC1C(F)F c1(C(=O)NCC(C(C)C)NC(=O)C=C2CCCCC2)cc2cc(Cl)sc2[nH]1 O(NC(=O)C(CCC1CCC1)NC(=O)CCc1cnn[nH]1)C(CC)C c1(CC)ccc(C(=O)C(=O)N(C2CCN(C(=O)CC=C(C)C)CC2)CCO)cc1 CCC(CCCC(=O)NCC1CC(SC)C1)NC(=O)CN(C1CCCC1)C CN1CCCC(NC(=O)C(C)(C)C(N)C2CCC2)CC1 n1(CC)ccc(C(N2CC(CC(=O)NC3CC(=O)N(C(C)C)C3)CC2C)=O)c1C CCCCS(=O)(=O)CC(=O)NC(C)(CNC(=O)C(C)OC)C(C)C C(=O)(C(C)C(C)C(C)(C)C)NCC12N(C(CNC(CC)=O)=O)C(CC1)CC2 N1(C(Cc2cn(CC)nc2)=O)CCN(C(=O)COCCN(C)C)CC1COC C1(NC(Cc2c(C)con2)=O)CN(C(c2nnc(O)cc2O)=O)CCC12CCC2 N1(CCC)CCCCCC1c1ccc(C)o1.C12CN(CC1CC1CC1)C(=O)N2C1CC1 N1(C(CNC(=O)OC)=O)C2CCC(C2)C1C(=O)NCc1cc(C)ns1 C1(NC(C(C2CN(CCCCN(C3CC3)CC)C2)OC)=O)CCSCC1 N1(C(c2ccc(C(C)=O)c(F)c2)=O)CC2CCC(C1)N2C(C1CC(C)(C)O1)=O N1(C(c2c(C)noc2C2CC2)=O)CCOCC(NC(=O)CC2(C)CCC2)C1 C1(OC(C(=O)OC)C)CCN(C(CCC2CCCCC2)C(=O)NC)CC1 C=CCC(CNC(c1cc(CC)ns1)=O)NC(c1c[nH]nc1OCC(F)F)=O c1(C(=O)NC(CCNC(C2=CC(C)(CC)C2)=O)(C)C)cc2c(o1)CCCC2 C1(C(=O)NC2(C)CCN(C(Cc3cccc(C)c3)=O)CC2)CCC2CCC(=O)N12 C1(CC(=O)NCC2CC(CNC(C3CCCC34CC4)=O)C2)CCCCCO1 N1(C(CC(C(C)C)NC(=O)C(C2CCOCC2)C)=O)CCC12CCN(C)C2 N1(C(C2CC(=C)C2)=O)CC(F)CC1C(=O)Nc1cnc[nH]1 C1(NC(C2CCC(C)O2)=O)CC2CCC1CC2NC(c1cc2ncccc2s1)=O C(=O)(CC(O)C(C)(C)C)NC1CC(CNC(C2CCC(=C)CC2)=O)N(C(C)=O)C1 C(CC(O)C(=O)NCC1CC1NC(=O)CCS(C)(=O)=O)SC C(=O)(CCCCCS(N)(=O)=O)NCC1C(NC(=O)COc2ccsn2)CC1 C1(OC)CC(CCNC(c2nn(C)cc2Cl)=O)N(C(=O)C(=O)N(C)C)C1.C(=O)C c1(CC)nnc(=NCCC(C)(C)NC(c2cnc3c(F)cccn23)=O)[nH]c1CC N1(C(c2ccc(C)cn2)C(=O)N2CCC2C2CCCC2)CC2CC1CS2(=O)=O C1(C(=O)OCC)CCCN(C(C2CN(c3ccccc3)C2)=O)C1 c1(C(=O)NC2CN(C(C34C(C)OC(CO)(C3)C4)=O)CC2C)cccc2nncn12 CC1(C(N2CCC(O)C(O)C2)=O)CCCN(C(c2ncsc2Br)=O)C1 N1(C(C(CC)N(C)C)=O)CCC(C)CC1CNC(C1(C)CC=CC1)=O CC(C)CCC(C(=O)NC1CN2CCC1(F)CC2)NC(C1CCOCC1)=O c1(C(N(C2C(N(C(CCCC)=O)C)CCCC2)C)=O)n[nH]c2c1CC1CC21 N1(C)S(=O)(=O)N(C)CCC1=O.CC1CC1 C(=O)(C(C)C(C)O)NCCN(C(CNC(c1c(C)occ1)=O)=O)CC1CC1 c1(C(=O)NC(CCCNC(C(c2scc(C)n2)C)=O)(C)C)coc(S(C)(=O)=O)c1 C1(NC(c2c(CC)onc2)=O)CCSC12CN(C(c1ccc3ncnn3c1)=O)C2 C(CNC(=O)C(C)(C)C1CCC1)(CC(=O)NCC1(F)CCC1)OC C1(NC(C(CSC)O)=O)CCCCC1CC(=O)NC1COCCOC1 C(CCCC(=O)N1CC2C(CNC(=O)C=CCN3CC4CCC3C4)C2C1)N(C)C Cc1sc(C(=O)NC(C)CC(C)NC(=O)C(F)CC2CCOC2)cc1[N+](=O)[O-] C1(C(=O)NCc2nc(C(C)C)on2)CCOCCN1C(c1cnc(Cl)s1)=O c1(-c2n(C)ncc2)cn(C)c2ccccc12.C(=O)(C)N(C1CCC1)CCN c1(N2CCCC(CC)C2)nc(N2CCCC(c3cncn3C)C2)cc(C)n1 n1(CC)nccc(NC(=O)C(N2CCCCC2CS(N)(=O)=O)=O)c1=O CC(CNC(C1SCCS1)=O)C(=O)NCc1nncn1C1CC1 C1(C(=O)NCC2(OC)CN(c3c(C)c(Cl)ncn3)C2)CCc2c[nH]nc2C1 C1(CNC(CC2CN(C)C2)=O)CCCN(c2cc(=O)n(C)cn2)CC1 C(C)(C(=O)NCCCN(C(=O)CN1CCC1C)C1CC1)OCC CC(C(=O)NC1CC2C(NC(=O)C(c3cccc(Cl)c3)O)C2C1)C(F)F Cc1ncsc1C=CC(=O)NC1CN(C(=O)CC2(n3ccnc3)CC2)CC1C c1(C(N(CC(F)F)C)=O)c(NC(=O)C(F)(F)C(F)(F)F)sc2c1CCCC2 c1(C(=O)NCC2CC3(CN(C(c4[nH]n(C)c(=O)n4)=O)C3)C2)cc2c([nH]1)CCOC2 C(CC(O)CO)N(C)C(C1(NC(=O)C(c2ccccc2)F)CC1(C)C)=O CCCCCCOCC(=O)NCc1csc(CNC(C2CCCN2CC)=O)n1 c1(CCN2CCN(CCC(=O)OC)C2=O)nc2ccccc2o1 c1(C(N(CCCN(C(CN(C)C(N)=O)=O)C)C)=O)nc(Br)n2ccccc12 CC1CCCC(C(=O)N(C)CC2CCN(C(=O)CCN3CCOCC3=O)CC2)C1 CN1CCC(C(N2CCC(CCNC(=O)C(C)(C)c3ccno3)C2)=O)CC1=O c1(-c2nc(C)c(NC(c3c(C(F)(F)F)cccc3F)=O)s2)ccc2c(c1)CCO2 C1(CCC)CCCN(C(C2CC(N(C)C(C3(NC(C)=O)CC3)=O)C2)=O)C1 c1(N(C(=O)COc2ccon2)C(C2C(C(N)=O)CC2)=O)nc(O)nc(O)n1 c1cccc(S(=O)(=O)OCC)c1.C1(NC(COCCOCC)=O)C=CC(C(=O)N)C1 C1(C(N2CC3C(NC(CSc4n(C)cnn4)=O)C(C3)C2)=O)C2CCCCCCC12 c1(C(=O)NC(CNC(CC(C(C)C)C)=O)(C)C2CC2)nnc(O)c2c1CCCC2 N1(C(C2C(NC(c3cnn(C(C)C)n3)=O)CC=CC2)=O)CC(C)(C)C12CCC2 C(CC(C)(C)C(=O)NCC1CCOC1=O)NC(CC1(C)CCCCC1)=O C(=O)(C(=O)C(C)(C)C)NCCC1N(C(c2nc(C)n(C)c2)=O)CCC1 C1(N2CC(OCC)C2)CCC12CCN(C(=O)OC(C)(C)C)CC2 c1(CCCC)ccc(S(=O)(=O)NC2CN(Cc3ccc(O)c(F)c3)C2)cc1 N1(C(CN2CCN(CC)CC2)=O)CCCC12CCCN(C(=O)C1=C(Cl)CCC1)C2 CN1C(=O)CN(C(C2CCN(C(C)(C)C)CC2)=O)Cc2ccccc21 C(=O)(CCCCC(=O)N1CCC2(C1)CN(C(c1cnc(S)nc1)=O)C2)NC N1(C(c2c(C)noc2N)=O)CC2CCC1C(NC(=O)C(N1CCCC(C)C1)=O)C2 c1(C(C)=O)cncc(C(=O)NC2(C)CN(C(=O)C(C)n3cccn3)C2)c1 C1(NC(C(CC)(C)C)=O)CC2CCC(C1)N2C(=O)CC1CCSCC1 C1(C(=O)NCC=CC(=O)NCC(CC=C)(C)C)OCCCC1(C)C C(=O)(CC(F)(F)C(F)(F)F)N(CCCCNC(C1CC2(CCCC2)CO1)=O)C C1(NC(C2CCCC23CCC3)=O)CC2COCC(C1)N2C(=O)CN1CC(F)(F)C1 C1(C(=O)NC2(C3CN(C(c4n(C)ccc4)=O)C3)CC2)Cc2ccncc2C1 c1(C(N(CC(CN(C(CCCSC)=O)C)O)C)=O)cccc2c1OCC2C c1(OCC)c(C)cc(C(C)NC(=O)N(CC(=O)O)CCO)cc1C C1(CNC(=O)C=Cc2cnc[nH]2)CC2(CO1)CN(c1c(Cl)cncc1[N+](=O)[O-])C2 C1(C#N)(C(N(CCNC(c2coc(Cl)n2)=O)CC)=O)CCCCC1 c1(C(=O)NCCC(=C)CNC(=O)CCC2CC(C)C2)cccnc1NC(C)C C1(OC)CC2CC1CN(C(C1CCN(C(=O)C3=CCCCO3)C(C)(C)C1)=O)C2 C1(CNC(c2scc(C)c2C)=O)CN(C(c2ccns2)=O)CCCO1 C1(n2cc(-c3cc(SC)no3)nn2)CN(C(=O)C(N2CCN(C)C2=O)C)CC1O C=CC(C)(C)CC(=O)N1CC2CC2(NC(=O)C(C)S(C)(=O)=O)C1.c12cccc(c1)S2 N1(C(C2(C)C=CCC2)=O)CCC2CCC(C1)N2CC1CC(F)(F)C1 c1(C(c2nnnn2C(C)(C)C)NC(CC=C)C2CC2)ccc(OC(F)F)c(Cl)c1 Cc1cc(C(N2C(CC(=O)NC3CCN(C)C(C)C3)C3CCCC23)=O)cc(C)c1 C(CC(=O)N(C)CCC1CC1)(C(F)F)NC(C(C)N(C(C)=O)C)=O n1(CC)cc(C(=O)NC2(CNC(c3sc(C)cc3C)=O)CC2)c(C)n1 N(C(=NCCc1ccccc1Br)NCC1CC1C)CC(F)=C(C)C N1(C(c2ncn(CC)n2)=O)CCCC2(C1)CN(C(C1CC(C)CO1)=O)C2 Cc1cc(Cl)nn1CC(=O)Nc1ccc(C(=O)Nc2c[nH]nc2Br)nc1 C1(c2n(CCCOC)nnn2)(NCCC2(C)COC2)CC2CC1CC2(C)OC N12CC3CCCC(C3C1)NC(=O)C1C(C1)C2=O.c1(C(=O)OC)n[nH]cc1OC c1(OC)ccnc(Cl)c1NC(=O)CNCCCCNC(=O)OC(C)(C)C c1(C(N2CCOCC(CNC(C3CCC(CC)O3)=O)C2)=O)scc2c1OCCO2 CCCC(C)(O)C(=O)NC1COCCN(C(=O)C=C2CCC(C)C2)C1 C1(CC(=O)NC(COC)CCO)CCN(C(=O)C(C#N)C(C)C)C1(C)C c1(SC)ccc(N)cc1C(=O)N(C1CCCC(NC(=O)Cc2ccoc2)C1)C CC1(C)C2CCC(C2)C1(C)C(N1CC(NC(c2cn(C3CC3)cn2)=O)C1)=O c1(C(=O)NC(C)CC2CN(C(=O)C(C)(F)F)C2)cscc1S(C)(=O)=O C1(NC(=O)CC2COCC2O)CN(C(c2cc(O)cc(O)n2)=O)C2(CCC2)C1 c1(OCC)cnc(C(=O)NCC2CN(C(c3ccc(CO)cc3)=O)C3CC23)cn1 C=C(C)CCC(=O)N1CC(O)CC1CNC(C1(C(F)(F)F)CCCCO1)=O c1(CN2CC(CC(=O)NOCc3cscn3)OCC2)c[nH]c2ccccc12 C12(C(=O)NCCC3(O)CN(C(c4ccc(F)c(Cl)c4)=O)C3)CCCCC1C2(F)F c1(N2CCN(c3ncc(C)s3)CC2)[nH]c(=NC2CCOC(C)(C)C2)nc2scnc12 N1(C(=O)CCc2ccon2)CCCC(NC(C2CC(Oc3ccccc3)C2)=O)C1 c1(CNCC(=O)OC(c2ccc(C)nc2)=O)cc(C)n(-c2ccc(Cl)cc2)c1C C1(CC)CC(C)CN(C(C2CCOCC2NC(=O)CCCc2ncco2)=O)C1 N1(C(c2ccc(SC)s2)=O)CCN(C(=O)CC=C(C)C)CC1CC(F)F N1(C(c2c(C)ncs2)=O)CC(CNC(=O)CC(=O)Nc2nccs2)CC1C C(CCC(F)(F)F)ONC(=O)C1CC1NC(C(C)CC1CCC1)=O N1(C(C(C)OCC(F)(F)F)=O)CC2(CCN2C(c2cncn2C)=O)C1 N1(C(C(COC)COC)=O)CC2(CCCC2NC(c2cc3sccc3n2C)=O)C1 CCC(C)(C)C(C)CC(=O)NCC(C1CC1)N(C(=O)CSc1ccc(F)cc1)C C(=O)(CS(=O)(=O)Cc1cccs1)NC1C(OC)CN(C(C(CC)=CCCC)=O)C1 Cc1ccccc1CCCNC(N1CC(NC(=O)OC(C)(C)C)CC1C)=O CCCC(C)CC(=O)N1CCC(C(=O)NCCN2CCC2)C1 C(=O)(C(C)C(CC)CC)N(CC(CC)NC(c1cnn(C(F)F)c1)=O)C C1(C(=O)NCC2(NC(C(N)=O)=O)CCC2)CCC(C(N)=O)CC1 C12(C(N(C3CCOCC3)C)=O)CC(CO1)N(C(C1CC3CCCC3C1)=O)C2 N#Cc1ccc(SCC(=O)Nc2cc(C(=O)O)nc(Cl)c2)cc1 c1(CNC(C2CCC(NC(c3c(CC)cccn3)=O)C2)=O)cnc(O)nc1O CC1CCOCC1C(=O)NCC1(F)CN(C(=O)Cc2ccc(C(=O)O)s2)C1 CCC(CCC(=O)NCC1C2CN(C(=O)C(c3ccc(F)cc3)C)CC12)OC C1(c2cc(C)[nH]n2)CCN(C(=O)CC2(C)CC2(F)Cl)CC1 N1(C(c2n3c(nn2)SC(=C)C3)=O)CCCC(C2CN(C(C3CCOC3)=O)C2)C1 c1(N(CC(=O)NCCC)C)nc(=NCC2CCCCC2O)[nH]c2ncn(C)c12 C(C)(C)(CCCNC(C1(O)CCC1)=O)NC(c1c(C)ocn1)=O C12(OC)CCC(C(=O)NC3CCN(CC(C4CC4C(F)F)=O)CC3)(CC1)C2 c1(CNC(c2cccc(NC(Cc3nc(=N)[nH][nH]3)=O)c2)=O)ccc(F)cc1Br N1(C(CC(C)n2cccn2)=O)CCCN(C(c2c[nH]ccc2=O)=O)C(CO)C1 C1(C(=O)NCC2CNC(=O)C2)(CC)CCCN1C(=O)CC1CCCO1 N#Cc1ccc(C(=O)NC23CC(C(=O)NCCOc4ccccc4)(C2)C3)s1 c1(C(=O)NC2CCN(C(CC=CCC)=O)C2)c(C)ncnc1C C(=O)(C(F)CC(C)(C)C)N1CC(NC(C)(C)C)C(C)(NC(=O)OC(C)(C)C)C1 N1(C(CCC=CC)=O)CC2OCCN(C(C3CN(S(=O)(=O)C(F)(F)F)C3)=O)C2C1 C12(C(N3C(CC(=O)N(C)CCN4CCCC4)CC(O)C3)=O)CCCN(CC1)C2 N1(Cc2ncc(OC)nc2)CC2CN(C(c3c(O)cccc3F)=O)CC2C1 CC(C)CCCC(C)(O)C(=O)NCCCC(CC)CC(=O)O c12cc(nn1CC)CC2=O.C1(CCOC)(C(=O)NC2CN(C3CC3)C2)CC1(F)F.C1CC1 N1(C(CS(=O)(=O)NC)=O)C2CCC1CN(C(c1ccc(OC)cc1COC)=O)C2 N#Cc1cc(C(=O)NC2CCC(CC(=O)NCCOCCOCCO)C2)on1 C(=O)(CCC(CC)NC(=O)CCCC1CC1C)N(CCCN(C)C)CCC C1(C(=O)NC2CC(CCn3cc(-c4c(C)nn(C)c4)nn3)C2)CC2(CCC2)CO1 N(C(=NCC(C)C(=O)NC)NCC(C)(O)c1cccs1)C(CC)CC CC(C(=O)NCC1CN(C(C23CCC2C3)=O)C1)(C(F)F)c1ccccc1 N1(C(CCC(C)OCC)=O)CCC(C2CCN(C(=O)Cc3ccn(C)n3)CC2)C1 Cc1cc(C(N2CCC(F)CC2C(N2CCN(C(C)C)C(=O)C2)=O)=O)cc(C)c1 C1(C(=O)OC)CCC(C(N2CCCC2CN(C)C(c2nc(Cl)cs2)=O)=O)C1 CC(C)(C)C1=NOC(C)(C(=O)NCc2cccc(CO)c2)C1.C12CCC1NC2=O CC(C)C(C)C(CNC(=O)CN1CCCC1)NC(C1(C(C)C)CCOCC1)=O Cc1cccc(C(O)C(=O)NC(C2CN(C(=O)Cn3ncc(Cl)c3C)C2)C)c1 C1(CNC(C(CCOC)(C)C)=O)CC2(CCN(C(c3coc(SC)c3)=O)C2)CO1 c1(OC)cc(C(=O)NC2CCOCC2C(=O)Nc2ccc(O)cc2Cl)ccc1C Cc1cc(C)c(CC(=O)NCCNC(=O)C2=COCC2)c(C)c1 c1(CN(C(=O)COCCF)C)cccc(CNC(C2CCC(=O)N2)=O)c1 N1(C(CCCC#CC)=O)CC(C(=O)NC(c2ncn(C)n2)C)CC(C)(C)C1 CCC(CCOC)C(=O)NC1CCN(C(=O)C(F)(F)C2CC2)CC1O C(=O)(CCCCCC(=O)NCC1CC1CNC(=O)C(C)(C)CCSC)OCC C1(C(=O)NC(C(=O)NCCCCCC#C)C2CCCO2)CC(C)N(C)C1 c1(C(=O)NC(Cc2cn(CCCOC)nn2)CC(=O)O)cc(F)cc([N+](=O)[O-])c1 Cc1noc(C(F)(F)F)c1C(=O)N(C1CCN(C2CC2)C1)C c1(CCC(=O)NCC2CCCC(NC(C3C4COCC34)=O)C2)ccc(F)c(Cl)c1 C#CCC(CC(=O)N1CCCC1CCO)NC(=O)C(C)(C)CCC N1(C(CC(=C=C)C)=O)CCN(C(c2ncc(Cl)cc2Cl)=O)C2CC12 C(=O)(C1Cc2ccccc21)N1CCC(OCCN(C(=O)CC2(C)CC2)CCOC)C1 c1(C(C)(C)C)ncc(C=CC(=O)NCC2(CNC(c3ccc(O)nn3)=O)CC2)s1 CCCCC(C(=O)N(C(c1ccccc1)C)CC)C(C)C.CCCCCCCCO Cc1ccc(O)c(NC(=O)CCc2ccc(NC(=O)CN3CCN(C)CC3)[nH]2)n1 C(=O)(C1=C(C)N(C)c2ncnn2C1)NC1CN(C(C(CC)(C)COC)=O)CC1O c1(C(=O)NCC2C(C(=O)NCC(=O)NCCC)CCC2)cc(C)ncc1C c1(C(N2CC(C)(CNC(C(CC)OCC)=O)C2)=O)ccc2c(c1)CCC(=O)N2 c1(OCOC)cc2ccc1CNc1ccc-2nc1C.c1(OC)nccc(C)n1 C12(CNC(c3scc(COC)c3)=O)CC1CN(C(C1(OC)CCSCC1)=O)C2 CCC(CC)(CO)C(=O)N1CCN(C(C2COCC(C)O2)=O)CC(O)C1 C1(CNC(C(C)CC(F)F)=O)CC2(CCC(CN)OC2)C1.C(=O)C(C)(C)C c1(C(=O)NCC2(C)CCN(C(c3cnc(C)s3)=O)C2)ccc2nc[nH]c2c1 C1(NC(=O)CCC2CCCO2)COC2C(NC(c3cccc(CO)c3)=O)COC12 C1(CCN2CC(C)(NC(C(CCSC)NC(C)=O)=O)C2)CCCCCCC1 Cc1nccn1CCCC(=O)NC(C)(C)CCNC(=O)C(C)Cc1ccco1 c1(C(N(CCC)CCNC(=O)C(F)CC2CC2)=O)cncc(C(N)=O)c1 C1(C)(CNC(C2(C)ON=C(C)C2)=O)CCCN(C(c2ccc(C)c(O)c2)=O)C1 C1(C(=O)NC2CC(CNC(c3sccc3C3CC3)=O)C2)CCCC2CCCN12 C1(C)(C(N2CC(C)C(NC(c3cnc4n3CCC4)=O)C2)=O)COC(=O)OC1 c1(C(=O)NC2(C)CCN(C(c3cc(C(C)=O)oc3)=O)C2)c2ccccc2nn1C c1(C(N2C(C)CC(CNC(=O)C(C)(C)C3CC3)C2)=O)ccc2nc[nH]c2c1 c1(CNC(C2CCSCC2)=O)ccc(CNC(c2ncoc2C2CC2)=O)cc1 C1(C)(NC(CC2CC(=C)C2)=O)CC(NC(c2ccc(CCCCCC)s2)=O)C1 c1(C(N2CCC(CC(N3CCC3CO)=O)CC2)=O)cc([N+](=O)[O-])c(Cl)cc1Cl N1(C(C2C=CCC2)=O)CCCC(N=c2[nH]c3ccc(O)cc3s2)CC1 N1(C(CSc2ccc(C)cc2)=O)CCC(NC(=O)CC2CSCCS2)C(O)C1 c1(C(N(CC(C(=O)NC(CC(C)C)C)C)C)=O)cc2ccccn2n1 c1(C(=O)NC2CCN(C(C3CC3c3cn[nH]c3)=O)C2)cc(Cl)c(F)c(Cl)c1 c1(CC)cccc(CN(C(=O)C(N)c2cncs2)C2CCC2)c1 C1(c2scc(C(=O)O)n2)CCCN(C(=O)CCc2nc(Br)cs2)C1 CC(C)C(C)(C)C(=O)NCCC1(C)CCN(C(=O)CCCN(C)C)C1 CC1(C)CCN(C(C2CCOC2)=O)CC1C(=O)NCCN=S(C)(C)=O CCCCCCC(O)CCC(=O)N1CC=CC1.C1C2CC3CN(C(=O)CC)C1C3C2 C1(Nc2cccc(CNC(c3nc(OC)sc3)=O)c2)Cc2cccc(OC)c2O1 C#CCC(O)C(=O)N(C1CN(C(=O)Cc2ccc(Cl)cc2)CC1O)C n1(CC(N2CCC(Nc3ccc(C)cc3)C(C)C2)=O)cnc2c1CCCC2 N1(C(c2c(C)cn(C)n2)=O)CC2CCC(C1)N2C(c1sc2cncn2c1C)=O N1(C(CSCCC(C)C)=O)CC2(CNC(c3nocc3Cl)=O)CCC1CC2 C1(C)(CNC(c2cn(C)nc2O)=O)CN(C(c2c[nH]c(=N)o2)=O)C(C)(C)C1 c1(C(=O)NCC2N(C(C(c3cn(C)nc3)O)=O)CC2)cccc(=O)n1O Cc1cc(Cl)c(C(=O)NC2CC(C)N(C(=O)C=Cc3ccccn3)C2)cc1C n1(CC)nc(C2CC2)cc1C(=O)NC1CC(CNC(=O)CCCc2cnn[nH]2)C1 Cc1cc(NC(C2CCN(C(=O)C3=CCC(C)CC3)C2)C)n2ncc(C)c2n1 c12ccc(o1)[nH]c2=O.N1(C(c2nccs2)=O)CCC(Oc2ccccc2)C1 c1(C(=O)NCC(C)NC(=O)C(C2(O)CCCC2)F)cc(Cl)c(C(F)F)cc1F N1(C(C(COC)NC(=O)CCCN(C)C)=O)CCCC(N=[N+]=[N-])CC1 c1(CN2C(C(=O)NCCc3nn[nH]n3)CC(F)C2)cn2cccnc2n1 CC1(C)CCCN(C(C2(C#N)CCOC2)=O)C1CNC(=O)COC1CC=CC1 C(=O)(C(C)C(O)C(C)C)N1CC(SC)C(NC(=O)CCc2nnc(C(C)C)o2)C1 C(=O)(C(F)COC)N1CC(OCC)C1.c1(C2C(=O)N2)ccnn1C CC1CN(C(=O)CC2CCN(C(=O)C3=CCCCC3C)C2)Cc2c[nH]nc21 N1(C(c2c(C)cccc2)=O)CCC2CCCN(C(c3cnn4ccsc34)=O)C2C1 CN1Cc2ccc(C(N3CCC4CC4CC3)C(=O)NCc3cccs3)cc2C1=O c1(NCCCN(C)C2CC2)cc(Br)ccc1S(=O)(=O)NCc1c(C)nn(C)c1Br C1(C(=O)NCC(CNC(CCC(=O)NCCC)=O)C)CC(=O)CC(=O)C1 Cn1[nH]c(C(N2CCC(c3cc(CNC(c4nccs4)=O)on3)CC2)=O)nc1=O C1(CC)CCC(C(=O)NCCCOCCC(=O)NC23CCCCC2C3)CC1 C1(OC)CC(c2ncc[nH]2)N(C(c2ccco2)=O)C1 c1(C(=O)NCC2CCCN(C(c3ccnc(O)c3)=O)CC2)cc2cccnn2c1 C(=O)(CCCC(C)O)O.C(CC(=O)NOC1CCCN(S(=O)(=O)C)C1)c1onc(C)n1 C12(NC(c3cc(C)on3)=O)CCCC(NC(=O)CC(C)(C)C3CCCCC3)(C1)C2 CC1CN(C(=O)C=CC(F)(F)F)CCC1NC(=O)C(C)(C)C C1(CC(=O)NC(C)CC(C)(C)C)(NC(C(n2ncc(C)c2)C)=O)CCCCC1 C1(C(=O)NCCC(CNC(c2nn(C)c(F)c2)=O)(C)C)CC(C)(C)OC1(C)C C1(CNC(CCCCN(C)C)=O)CN(C(C2CCCN2C)=O)CC2(CCC2)O1 Cc1c(C(N2CCC2C(=O)Nc2ncc(C#N)cc2Br)=O)cc(F)cc1[N+](=O)[O-] Cc1cccnc1C=CC(=O)NCC1(CN(C(=O)CC2CC2C)C)CC1 C1(C)(CNC(C(C)OCCCC)=O)CCCN1C(c1ccc(SC)o1)=O CCC(CC(F)(F)F)C(=O)N1CCCCC1CNC(=O)CNC(N)=O C1(O)(CN(C(CSCC#C)=O)C)CCCN(C(c2cc(C(=O)OC)nn2C)=O)C1 C1(NC(=O)CC2CCCSC2)CC2C(NC(c3cnc(O)o3)=O)C2C1 C1(NC(CCOC(CC(C)C)C)=O)CN(C(c2cc(C3CC3)ns2)=O)CC1(C)C c1(C(=O)NC2CCCN(C(CC3CC(NC(C)=O)C3)=O)C2)ccc(N)c(Cl)n1 C1(CNC(Cn2ncc(C)c2)=O)CCC(C)CN1C(=O)CC1(N(C)C)CCCC1 c1(C(=O)NCCCN2CCOCC2)nsc2cc(-c3ccccc3F)ccc12 N(C1CC(C)n2ccnc21)C(C12CN(C(c3cc(=NC)[nH]cc3)=O)C(C1)CO2)=O C1(CNC(c2cc(F)cs2)=O)C2CN(C(=O)C3=COCC3)CC12 c1(C(=O)NC(CNC(c2c(C)cns2)=O)CC(C)C)ccc2c(c1)C(C)(C)CN2 CC(C(C)(C)C(=O)N1CCC(F)(F)C1)NC(C1CCC(N(C)C)C1)=O N1(C(C(C(CC)C)OC)=O)CCC2(CC(NC(C3(S(N)(=O)=O)CC3)=O)C2)C1 C(=O)(CC(C)C(F)F)NC(C1CN(C(C(N2CCC(C)CC2)=O)=O)C1)C c1(C(=O)NC(C)CCCCNC(=O)CNC(=O)CO)ccnc(O)c1Br c1(C(N2CCCCC(NC(CN3CCC(C)CC3)=O)C2)=O)cc2c([nH]1)CCCC2 N1(C(CC2CC(C(C)C)OCC2)=O)CC2(CNC(C3CC(O)C3)=O)CCC1CC2 n1(CC)nc(-c2ccc(C)cc2)nc1-c1cccnn1 C1(C(=O)NCc2ccc(C)c(C)c2)CC12CCN(Cc1ccc(Br)[nH]1)CC2 c1(C(=O)NC(CC=C)CNC(c2c(C)[nH]c(C)c2C)=O)csc(=NC2CC2)[nH]1 CC(C)CCC(C(=O)N1CC2(CCCO2)C1)NC(C1CC2CCCC2C1)=O C(=O)(C1=CCCCC1)N(C1CCN(C(c2cnn[nH]2)=O)CC1)C C1(CNC(C(C#C)(C)C)=O)CCC2(CCN(C(=O)CN(C)CC)CC2)CO1 c1(C(=O)NC(CCC)C(=O)NC2CCCN(c3ncccn3)C2)cc2n(n1)CCO2 C(=O)(C(C#N)C(C)(C)C)NCC(CC(=O)N1CC(NC(COC)=O)C1)O C(=O)(C1=C(Cl)CCOC1)NCCN(C(C1CCCC(C)(C)C1)=O)Cc1ccccc1 C(CC(C(C)(C)C)NC(c1cnn(C)c1Cl)=O)N(C(c1c(C)cc(F)s1)=O)C c1(OC)c(C(=O)NC2(C)CCN(C(c3cc(C)oc3C)=O)C2)csc1Cl C1(CNC(C2CC(F)(CNC(C3(CC)CCC3)=O)C2)=O)CC12CCOC2 c1(C(=O)NC(C)CN(C)C(c2cnns2)=O)cn2cccnc2n1 C1(CNC(C(CSC)O)=O)CCCCCN1C(=O)C#CC1CC1 c1(OCC)cccc2cc(CN(C3CCC(NC(=O)NCC)CC3)C=O)oc12 CC(F)(CNC(=O)C1CC1)CNC(C1(C)CC1(Cl)Cl)=O N(C(=NCC1CCCC(C)(C)C1)N1CC(O)C2(CC2)C1)CC(C)C c1(OC)cc(CCn2nnnc2C2(NC(C)CC(C)C)CCSCC2)cc(C)c1 Cc1cccc(OCC(=O)NCCO)c1C.C(=O)(C(O)C1CCCC1)NCCCS CC(CCNC(=O)CCCCN1CCCC1)CCNC(C1CCCC1C)=O CC(C)CC(CN(C)C)NC(=O)C(O)CNC(C1CN2CCC1C2)=O N1(C(c2cc(C(C)=O)on2)=O)CCC(CN(C)C(C2(C)CCSCC2)=O)CC1 CC(C)C(O)C(=O)N(C(C)CNC(=O)CCCc1ccc(C(C)(C)C)cc1)C N=c1nc[nH]n1CC(=O)NC1CCOC1C(=O)NCCCSC(F)F C1(C(=O)OC)(CF)CCN(C(=O)C(=O)NCCCC2COCCO2)C1 C1(C(C)NC(=O)C(C)(C)CF)CCN(CC2CCC(c3ccccc3)C2)C1(C)C c1(C(N2C(C)CCN(C(c3ncccn3)=O)CC2)=O)noc2c(F)cccc12 C1(NC(C2(C(C)C)CCC2)=O)CC2CCC1C(NC(c1cnns1)=O)C2 N1(C(c2cc(COC)sc2)=O)CCC(CCCNC(c2cccc(=O)o2)=O)CC1 C(=O)(C(CO)C(F)(F)F)NCC(CC=C)C(=O)NCC1CCCC(C)C1 C1(CC(=O)NC(C(=O)N(CC(C(C)C)OC)C)C)CCCC(=O)C1 N1(C(COCC=C)=O)CCC(C(F)(F)F)CC1CNC(=O)CC1OCCCO1 C1(CCOC)(NC(C2CC2Cl)=O)CCN(C(c2cccc(C(C)C)n2)=O)C1 C1(CC#C)(C(=O)NC(CNC(=O)Cc2cccn2C)(CC)CC)CCOCC1 C=C(CNC(C1(O)CC(c2ccccc2)C1)=O)CCNC(=O)CSS(C)(=O)=O c1(NC(CC)=O)ccc(NC(C2CC(C)N(c3cc(OC)ncn3)C2)=O)cc1C N1(C(CC(=O)OC)C)CCC2CN(C(c3cccc4nn(C)nc34)=O)CC2C1 C1(C(N(C)Cc2ccccn2)=O)CN(C(c2ncc(F)cc2F)=O)CC(C)(C)C1 CC1C2=C(C(=O)N1C)C(c1cccc3ccnn13)NC(=S)N2CCF C(=O)(C(CCC)C(=O)OC)NCCOC1CCN(C(C2CCC(=C)CC2)=O)C1 c1(CC)cccnc1C(N1CCC(C)(NC(=O)C(C2CCC(=O)N2)C)C1)=O C1(CC)(NC(c2occ(C)c2C)=O)CCN(C(=O)CC2COCCO2)CC1 c1(-c2cn(C(C)=O)nc2)cccc2[nH]nc(C(N3CCC(O)C(C)C3)=O)c12 S(=O)(=O)(c1cc(C(=O)O)c(Br)cc1F)Nc1ccc(CCN(C)CC)o1 C(=O)(C#CC1CCCC1)N(C1C2CN(C(c3cc(F)cc(Cl)c3N)=O)CC12)C N1(C(C(C)O)=O)CCC2(C1)CN(C(c1c(F)ccnc1F)=O)CC(C)O2 C1(NC(C2CCN(C(CC)=O)C2)=O)CC(C)CN(C(c2cnc(C3CC3)o2)=O)C1 CC1CN(C(=O)COC2CCCCCC2C)CCC1C(=O)NC1CC=CC1 C1(OC)(CNC(C2CC3CCC2O3)=O)CCN(C(c2cnn(C(C)C)c2)=O)CC1 c1(CC(=O)NC(C(C)C)CCO)c(F)c(F)cc(F)c1F c1(C(=O)NC2CCC3(CN(C(CCN(C)C)=O)C3)C2)cc2cc(Br)ccn2n1 N1(C(COCC)=O)CC2(CCCC2CC(N2CCCC(F)C2)=O)C1 C1(NC(C2CN(C(C)C)C2)=O)CC2COCC(C1)C2NC(C1CC(C)(C)C1)=O N1(CCCNC(C2C(CNC(c3cc(CC)on3)=O)CCC2)=O)CCCOCC1 c1ccc(-n2cc(CCNCCCn3ccnc3)nn2)cc1 N1(C(C2CN(C(=O)NC)C2)=O)CC2(NC(c3ccnc(CO)c3)=O)CCC1CC2 O=Cc1sc(CN2CCCC(C(N3CC(O)C(F)C3)=O)C2)c(Br)c1Br c1(C2(C(N3CCN(Cc4ccccc4)CC3CO)=O)CC2)cc(F)cc(F)c1Br N1(C(C(CCC)(C)O)=O)CC2(CC(C(=O)NC3CC(CC(N)=O)C3)CO2)C1 c1(C(=O)NC(CCN(C(CC(CC)C2CCC2)=O)C)C)cccc2oc(C)nc12 Cc1oc2ccccc2c1C(=O)NC1CCC2(CCNC2)C1 N1(C(C(=C)F)=O)CCC2(CC(C(=O)Nc3cc(O)ccc3Br)=NO2)C1 C1(C(=O)NCCCC2C(C)C2)CC(NC(C2CN(C)C2)=O)C(O)C1 C(=O)(C(CC(C)(C)C)NC(=O)C#CC1(C)COC1)NC(C)CO C1(NC(C2(CCCC)CC2)=O)CCC2(CCCN2C(c2cc(C)on2)=O)CC1 C(=O)(C#CC1CN(C(=O)OC(C)(C)C)C1)N(C)CCN(C)C(C1(C)CC1(F)F)=O C(=O)(CC(C)C(C)(C)NC(C1C=CCCC1)=O)NC1C2(CC(OCC)C2)C1 Cc1cnc2cccc(C(=O)NC(C)(C)C(C)NC(=O)CCC(C)C)c2c1 Cc1cn2nnc(C(=O)NCC3(O)CN(C(C45CCC4C5)=O)C3)c2c(O)n1 C=CC1CCCN1C(c1csc(C2CC2)n1)C(=O)NCCCF C1(N(C)C(c2csnn2)=O)CCCC(NC(=O)COCc2ccnn2C)C1 C1(NC(C2(NC(c3[nH]c(=N)sc3)=O)CCCCC2)=O)CC2C(O)C(O)CC12 C(=O)(CC1=CCCC1)NCC(C1CCN(C(=O)CCCc2ccccc2)CC1)C Cc1cc(C)c(CNC(C2CCCCN2C(=O)NCc2cccnc2)=O)[nH]1 C(=O)(C1COc2ccc(F)cc21)N1CC(C(C)NC(c2c(O)ccc(C)n2)=O)C1 c1(C(N2CCC(O)(C(C)NC(C(F)OC)=O)C2)=O)cc(N)c(N)cc1F C1(CC)(NC(=O)C(C)N(C)C(c2nocc2C)=O)CC(C)C1 c1(C(N(CCN(C(C23CCC2C3)=O)CC)CC)=O)sc(C2CCOC2)nc1C C(=O)(CCCC(=O)NOC(C)(C)C)N1CC(NC(C(C(C)C)C)=O)C(C)CC1 N1(C(c2cnn3ccsc23)=O)CC(CO)C2(C1)CN(C(=O)C(F)(Cl)C1CC1)C2 Cc1ccc2occ(CC(=O)NCC(C3CC3)NC(C3CCOC(C)C3)=O)c2c1 c1(C(=O)NC(C(=O)NC2(CCOC)CC2)Cc2cn[nH]c2)cccc2c[nH]nc12 C=CCCC(CC(C)C)C(=O)N1CCC(C)(NC(c2ccc(CN(C)C)[nH]2)=O)C1 C1(C(N(CCNC(CSC)=O)CCOC)=O)CCC(C)=C(C)C1 c1(C(N(CC(C)O)CCNC(C23CC(O)C2C3)=O)=O)cn(C)nc1Br c1(C(=O)NC(C)CCNC(C2CC2C(F)(F)F)=O)cc(-c2ccccc2)on1 c1(C(C)C)conc1C(=O)NC1CCC1CNC(=O)C(C)Cc1ccncc1 c1(SC2CC(CO)C2)cn(CCNC(C2(F)CCOC2)=O)nn1.C1(CS)CCS1(=O)=O c1(OC)cc(NC(C)=O)cc(S(=O)(=O)N2CC(CO)OC(C)C2)c1 C1(N=c2nc3[nH][nH]cc-3c(O)n2)(CNC(c2c(C)ccc(C)n2)=O)CCC(C)C1 FC(F)(F)C(F)CNC(c1ccc(CC2CC2)s1)c1nnnn1CC(F)F N1(C(C(C=C)O)=O)CCN(C(c2c(C)nn(C)c2Br)=O)CC1C1CC1 Cn1ccc2ccnc(C(=O)NCC3(O)CCCN(Cc4cscn4)C3)c12 CC1CCN(C(=O)C(C2CCC2)C2CCC2)CC1CNC(c1ccccc1O)=O C1(CNC(C2C(C)C2C)=O)CCC2(CN(C(c3nccnc3N)=O)C2)O1 c1(NC)ccc(Cl)c(C(=O)NCC2(F)CCN(C(=O)CCC3CCC3)CC2)c1 C1(NC(C=COCC)=O)C2CN(C(=O)C(C)(C)OCC)CC12 CCCC(C(=O)NC1CC(NC(=O)Cn2nc(C)oc2=O)C1)N(C)C Cc1cc(CNC(=O)CC2(C)CCN(C(=O)CC3CCC(=O)NC3)C2)cc(O)n1 Cn1nccc1C(C(=O)NCCCc1cc[nH]n1)NC(=O)CC12CCCC1C2 N1(C(c2[nH]nnc2C)C(=O)NCC(=C)C)C2CCC1CC1(C2)N=N1 Cc1cc(C(N2CCC(C(C)NC(C34COCC3C4)=O)CC2)=O)cc(=O)n1C Nc1ccc(S(=O)(=O)NC2CCCCCC2)nc1.c12nc(no1)C1CCCN21 c1(C(N2CCN(CCNC(c3cnc(C)o3)=O)CC2)=O)cnn2ccn(C)c12 CC1CN(C(=O)C=CC2CCCCC2)CC1CC(=O)NCCc1ccccn1 c1(OC)cn(C)c(C(=O)NCC2C3CN(C(c4c[nH]nc4OC)=O)CC23)cc1=O c1(C(N2CCC(CNC(C3CC4(CC(=C)C4)C3)=O)CC2)=O)ccc(N=[N+]=[N-])cn1 C1(C(C)OC)CCC(NC(=O)NCC(C)(O)CSC)C1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC(C(N2CCC(C)(F)C2)=O)C1(C)C N1(C(c2ccc(OC(C)C)cn2)=O)CC2(C1)SCCC2NC(=O)C(O)CC(F)F c1(C(=O)NCC2(NC(=O)CC3CCC(F)(F)C3)CC2)cccc2c1CCS2(=O)=O c1(SC(C)(C)C)ccc(-c2nc(C3CCCCCC3)nn2C2CCS(=O)(=O)C2)cc1 C=CC1OCCC1C(N1CCN(C(C)CNC(=O)C(O)C2CC2)CC1)=O C1(CC)(CC)CN(CC(=O)NC2COC(C)(C)C2)CCO1 N1(C(C(C)CNC(=O)C(C)(C)N=[N+]=[N-])=O)CCC2(CNC(=O)C2)C1 C1(CNC(CCC(=O)NCC)=O)CN(C(C2C(C)C2C)=O)CCC12CCC2 N1(C(C(C(C)C)F)=O)C(C)CN(C(C2CC(F)(F)C2(C)C)=O)CC1C C(=O)(CCS(N)(=O)=O)N(C)CC1CCN(C(c2cc(CO)[nH]n2)=O)C1 C(=O)(NN1CCCC1C(=O)N(C1CCOCC1C)C)C1C(OC)C1(C)C C1(CSC)CC(N=c2nc(N3CC4C(C3)C4(C)C)c3sccc3[nH]2)C1 S(=O)(=O)(c1cnc(N2CCCC(CC(F)F)C2)cc1C)N(C(CCC)C)C c1(CC)nc(C)c(CNC(=O)C(C)NC(c2ccc(C)cc2)=O)o1 c1(C(C(=O)NCC(C)N(C(c2ccccc2)=O)CC)N(C)C)ccc(F)c(Cl)c1F C#Cc1cnn(C)c1C(N1CCCC(C(N2CC(CS(C)=O)C2)=O)CC1)=O N1(C(CCC2CCC(C)O2)=O)CCC(CNC(c2cccnn2)=O)C12CC2 C(C1CCC(C)CC1)=C(C)C(N1CCN(C(C2CCN(C)C2)=O)CC1)=O CC1OCCCC1C(=O)NC12CC(C1)N(C(=O)C(F)=C1CCC1)C2 C1(C(N(CC(C)N(C)C(c2csc3nnsc23)=O)C)=O)CCn2nncc2C1 CC(C)(F)C(C)(F)C(=O)NCC1CN(C(=O)CCc2ccccc2F)CC1O C(C(C)(C)CC(C)O)NC(C(CC1CCC1)NC(C=C(C)C)=O)=O C1(NC(c2cncc(CC)n2)=O)CCN(C(C2CC(C(=O)OC)C2)=O)C(C)C1 c1(CC(=O)NC(=O)NCC)cc(CC2CC2)no1 C(=O)(C1(C)CCc2ccccc21)N1CCCC(COC)(NC(=O)CCC(N)=O)C1 N1(C(c2cnc(C(C)OCC)s2)=O)CCN(C(=O)C(F)=CC2CC2)CCC1C C1(C(N2CCC(C)(N(C)CC)C2)=O)CCCN(C(=O)CCCN=[N+]=[N-])CC1 c1(CCC(=O)NC2(CNC(C3C(CC)CCO3)=O)CCOC2)cccc(F)c1F c1(N2C(C)CC(CNC(C(c3ccc(Cl)s3)C)=O)C2)ncnc(Cl)c1F C(C)(CCC(=O)N1CC(O)CC1C(N1CCC(c2ncco2)C1)=O)OCC CCCC(O)C(CO)NC(C1CC(CCNC(c2ccncc2Cl)=O)C1)=O C(CSC)(C(=O)N(C1CCN(C(=O)CCc2nccn2C)C1)C)OC Cc1cc(F)cnc1C(=O)NC1CCOC(C(=O)N(C)CCc2cnccn2)C1 c1(CNC(c2ccc(N(C)NC(CSC(C)C)=O)cc2)=O)ccc(N)cc1.CCF CC(C)C(C)C(=O)NC1CCCC1NC(=O)CCC1CC(C)(C)CO1 C(=O)(C1CCc2ccc(Cl)nc21)NCC(C)NC(c1cc(=O)n(C)o1)=O c1(C(=O)NC2CN(C(C(CC=C)CC)=O)CC2(C)C)cc2c(C)c(F)ccc2[nH]1 C1(n2cc(-c3cc(C)ns3)nn2)CC2CCC1(NC(c1ccc(C(N)=O)[nH]1)=O)C2 C1(C(N(CCC)CCC)=O)CCC1NC(=O)C(C1CC1)ON.CC C1(N=[N+]=[N-])(C(=O)NCc2c(C)csc2)CCN(C(=O)C=Cc2nccs2)C1 Cc1c(F)ccc(C(N2CCOCC(NC(C3(C)CC3Br)=O)C2)=O)c1N c1(N2CC(F)(C(=O)NCC3(O)CCOCC3)C2)ncnc2cc(Br)sc12 Nc1ccc(C(N2CC(NC(c3cnn(CCF)c3)=O)C2)=O)cc1F c1(CC)cccc(C(N2CCOC(CNC(C3(C)CC(O)CN3C)=O)C2)=O)c1O C(CCCCN=c1[nH]c(=NCCCSC)[nH]c2ccsc12)CC C1(C(=O)NC2(CC)CCC2)CCCN(C(C2(C(C)C)CC2)=O)CC1 c1(C(=O)NC(C(C)C)CCNC(C2CCCCC2)=O)cc(F)cc2cc[nH]c12 CCC(C(=O)OC)C(=O)NCC1(OC)CCN(C(=O)Cc2cnoc2)C1 CC1(C)C(NC(=O)CCOC2CCCC2)CC1CNC(=O)C=Cc1cncs1 c1(C(=O)NCC(C)N(C(=O)C=Cc2ccco2)C)ccc2c(c1)NC(=O)CS2 C1(C(=O)NCCC=CC(=O)N(CC#C)CCF)C(C(C)=O)C1(C)C N1(C(C2(C)CC=CCC2)=O)CCC(NC(C2CCOC(=O)N2)=O)C(CO)CC1 C(CC(C)C)(C(=O)NCCc1ccnn1C)N(C(C(=O)NCC)=O)C C1(C(N(CC(C)O)C2CC2)=O)CC2CC1CC2NC(c1ccc(C(N)=O)[nH]1)=O O=C(C1=CCSC1)NC1CCCCC1NC(c1c[nH]nc1-c1ccsc1)=O C(c1ccc(F)c(F)c1)=CC(N1CC(C(N)=O)(CNC(CCC(=O)NC)=O)C1)=O c1(OCC(=O)NCC2CCN(C(C3CS(=O)(=O)C3)=O)CC2)ccc(Cl)cc1Cl C1(C(=O)NC(CC)(C)CNC(=O)CC(C)c2ccco2)CN2CCCC1C2 N1(C(CC(CC)C)=O)CCN(c2nc(C(C)(C)C)nc(=N)[nH]2)CC(O)C1 C(N=c1[nH]ccnc1N1CCC(n2cc(Cl)cn2)C1)c1n(C)c(Br)nn1 c1(C(N)=O)cc(N2CCCC2CCCNC(c2ccc[nH]2)=O)nc(Cl)n1 CC(C)CCCC(=O)NCC1CCN(C(=O)CC2(O)CCN(C)CC2)CC1 N1(C(C(CC(C)=O)C)=O)CCCC2(CCCN(C(c3sccc3F)=O)C2)C1 c1(OC)cccc(CC(O)CCN2CCC(c3ncc[nH]3)C2)c1 CC(C)CC(CC(=O)NC1CCCC1C#N)NC(c1cc(C#N)ccc1N)=O N1(C(c2cnc(C)s2)=O)CCC2CCC(C1)N2C(=O)Nc1cccc([N+](=O)[O-])c1 C1(C)(OC)CC(NC(C2CCCN(C(=O)C3=CCSC3)CC2)=O)C1(C)C CC1CCN(Cc2csc(Br)c2)CC1NC(c1cnoc1-c1ccccc1)=O c12ccc-1cc2.c1(CCC(=O)N(CCCO)CCCO)nc(C2CCCC2)no1 CC1(C(=O)NCC2CC(F)CN2C(C2CC2F)=O)CCCCC1 C1(C)(CC(=O)NCc2onc(COC)n2)CCCN(C(=O)C(C)(C2CC2)OC)C1 N1(C(C=C(CC)C)=O)CCN(C(=O)C(F)C2CCCC2)CC1CF c1(C(=O)NCC(C)NC(=O)C(c2ccccc2)O)cncn1-c1ccccc1 C1(O)(CCNC(C2CC3C=CC2C3)=O)CCCN(C(C2(Cl)CC2)=O)C1 N1(C(c2cn(CCC)nc2)=O)CC(F)CC1C(N1CCCC(CCO)C1)=O c1(C(=O)OCC)ccc(F)c(C(=O)NC2CCC3COC2O3)c1 CCCCCCC(=O)N1CCOC(Cn2cc(CC(O)C(C)C)nn2)C1 O=C1OC2CCN(C(c3c[nH]c(-c4ccncc4)n3)=O)CC2O1 C(=O)(C(O)CC(C)(C)C)N(C)Cc1nnc(CC)o1.C1(=O)CC(C)(C)N1 N1(C(C2Cc3n(cc(C)n3)C2)=O)CCCC12CCN(C(=O)C(C)O)C2 c1(C(N2CC(CNC(C=C=C(C)C)=O)N(C)CC2)=O)cc(N)c(F)cc1C C1(CNC(C2CC2C2CCCCC2)=O)CN(C(=O)C=CCO)C2(CCOCC2)C1 N1(C(C2C(C)(C)CO2)=O)CC2(C1)CN(C(c1ccnc(SC(C)(C)C)c1)=O)C2 N1(C(CC2(C#N)CC2)=O)CCC(OCCNC(=O)CSc2cccc(Cl)c2)CC1 c1(N2CCCC(C(N3CCC(Br)CC3)=O)CC2)ncnc2cc(I)sc12 c1(NC(=O)CC2CCN(S(=O)(=O)CCc3ccccc3)C2)ccn2ccnc2c1 C1(C(=O)OCC)CCN(c2nnc(CC(C)(O)C3CC3)n2C(C)C)CC1(C)CC C(=O)(CS(=O)(=O)CCO)NC1C(NC(c2cnn(C)c2C(F)F)=O)CCC1 NS(=O)(=O)c1sccc1C(N1CCCC(NC(C23CC2COC32CCC2)=O)C1)=O Cc1cccc(OCC(=O)OC(C)C(N2CCSC(C)(C)C2)=O)c1C c1(C(N2C(C(=O)OC)COCC2)=O)cc(OC)c(O)cc1Br.C1(=O)C(C(C)O)N1 C1(C(C)(C)C)CC(N2CCC(CC3CCCCO3)C2)C(=O)O1 C(C1CN(C(=O)Nc2ccc3c(c2)CC(C)(C)O3)Cc2ccccc21)NC(C)=O CCC(CN(C)C)CC(=O)NCCC#N.c12nc(co1)C(=O)N(CCCO)C2 CC(CC(=O)NC1(C)CC(NC(=O)Cn2cccnc2=O)C1)C(F)(F)C(F)(F)F CN(OCc1ccccc1)C(=O)C1COCC1CCC(F)(F)F C=Cn1nccc1C(=O)NC(C)(C)C(=O)Nc1cccc(C(C)C)c1 N1(C(C2(C)CCCS2)=O)CCCC(O)(CNC(=O)Cn2cc(C(F)(F)F)cn2)C1 C(=O)(N=c1c(C)c[nH]cc1C)c1c(C)ccc(NC(C)=O)c1 c1(CC)cc(CC)nc(C(=O)OC)n1.C12(CCCCC1)C1(CC1)CNC2=O N1(C(C(C(=O)OC)C)=O)CCC2CN(C(c3cccc(Cl)c3F)=O)CC2C1 c1(C(N2CC(NC(C(=O)NC)=O)C(C)C2)=O)cc2cc(F)ccc2o1 CC1CCC(=CC(=O)N(C2CN(C(c3csc(-c4ncccn4)n3)=O)C2)C)CC1 Cc1ccc2c(C(=O)NC3(C)CCCN(C(c4sccc4F)=O)C3)ccnc2c1 C(C(CN=c1[nH]nc(O)s1)C(F)(F)F)NC(=O)C1CC1c1ccccc1 CS(=O)(=O)C1CN(C(c2ccc(Cl)cc2O)=O)C2(CCC2)C1 c1(CN(C(=O)CCNc2cccc(Br)c2)C)cc(S(N)(=O)=O)c(Br)s1 C1(N(C(C(C)SCCCC)=O)C)CCCCN(C(=O)C(C)(C)c2cnn(C)c2)C1 C1(C(=O)NCCCCC(CO)NC(Cc2c(C)scc2)=O)Cc2ccccc2O1 N1(C(C(C)SCCCC)=O)CC(O)(C2(CNC(C3CCCN3C(C)C)=O)CC2)C1 N1(C(=O)OC)C2CCC1CC(CNC(=O)C(C13CC(CO)(C1)OC3C)N(C)C)C2 N1(C(C2CCC(C)O2)=O)CCC(NC(c2occc2C2CC2)=O)C(F)C1 C12(C(N(CCOC)CCNC(=O)CSC)=O)CC(OC)C1C2 c1(CCCC)cc(C(=O)NC(C)CCNC(C2(CO)CC2)=O)c(C)o1 Cc1c(C(=O)NC2CCC2CNC(=O)C(C)OC2CCOC2)cnn1C C12(NC(c3cccc(C)n3)=O)CCCCC1CN(C(C1(N(C)C)CC1)=O)C2 c1(C(=O)NCCC2CC(NC(c3nc(C(C)(C)C)sc3)=O)C2)ncc(F)cn1 C(=O)(CCN=c1ccc(C#N)c[nH]1)NCC1C(NC(C(C(C)C)NC(C)=O)=O)CCC1 c1(NC(N2CC(OCCNC(C(C)(C)C3CCCO3)=O)C2)=O)ccc(O)c(Cl)c1 C1(CC(=O)NC2(CNC(C(C)=C3CCCC3)=O)CCOC2)CC(C)(C)CCCO1 c1(CN2C(C(=O)Nc3cc(OC)n[nH]3)CCC2)cc(C)n(-c2ccccc2)c1C c1(C(C)C)ncc2c(n1)CN(C(=O)C(N1CCC(c3cccc(F)c3)C1)=O)CC2 C1(NC(CNC=O)=O)CN(C(c2cnco2)=O)CC2(CC2)C1 C(CCC(C)(C)NC(=O)CN(S(C)(=O)=O)C)NC(CSCC#C)=O.C=O C1(NC(CCNC(COC)=O)=O)CN(C(c2cccc(CO)n2)=O)CC12CCC2 N1(C(C2C(C)C2)=O)CC(CNC(c2cccc(-c3cnn(C)c3)c2)=O)C(O)C1 C12(NC(CCc3cc(OC)c(Cl)cc3)=O)CCC(CN(C(c3cc[nH]c3)=O)C1)C2 N1(C(=O)NCCOc2ccccc2Cc2ccccc2)CCC(CC)C(F)(F)C1 c1(C(N2CCC(NC(CC=CCC)=O)C2)=O)nn(CC)nc1C C(C)(C(=O)Nc1ccc(-n2cnc(C(N)=O)n2)cc1)(C(F)(F)F)OC CC1CN(C(c2coc(Cl)n2)=O)CC(C)C1N=c1ccnc(CC2CC2)[nH]1 C(CCCC(=O)NCCCCCCN(C(=O)Cn1cnc(C(N)=O)n1)C)OCC c1(OC)ccc(F)cc1CN1CCC(C(c2ccccc2)=O)C1 N1(C(C(C)N(C(C)=O)C)=O)CCCC(F)(CNC(c2cc(C)nn2C)=O)C1 CC1(C)C(CNC(=O)CCC2CCN(C(C3(C#N)CCCO3)=O)C2)C1(F)F C1(CNC(C2(C)CC(C(F)(F)F)C2)=O)CCCCN1C(=O)CC1C=CCC1 C1(CCC(=O)N(CC(CC=C)O)C)CCCCN(C(C2CC(C)(C)CO2)=O)C1 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(CNC(C2(F)CCOC2)=O)C(C)(C)C1 c1(C(N2CC(c3n(C)cnc3)C(CNC(=O)C(N)=O)C2)=O)ccc2n[nH]cc2c1 c1(-c2ccc(C(F)F)o2)nc(C2CCCCC2)nn1-c1ccc(Cl)nc1 c1(OC)ccc(C(C2CCN(C(=O)CC3CCCN3C(C)C)C2)(C)O)cc1 CCCCC(F)(F)C(=O)N1CC(OC)C(C(=O)NC(c2ccns2)C)C1 C1(CNC(C2(CCC)CC2)=O)(CO)CCN(C(=O)CC2CCCCC2)CC1 C1(C(C)NC(=O)COCC(=O)OC)CCCN1C(c1sccc1OC(F)F)=O N1(C(=O)NCCC(=O)N(CCCCN(C)C(C2CC2F)=O)C)CCCCC1 c1(OC)cc2c(cc1NC(=O)C(=O)NCc1ccc3nonc3c1)CCC2 N1(C(Cc2c(C)occ2)=O)CCC2(NC(=O)CCn3cccn3)CCCC12 c1(C(=O)NCC=C2CCN(C(c3c(C)c[nH]c3)=O)CC2)cccc(Cl)c1F c1(C(N2CCC(OCCNC(=O)CSc3nncs3)C2)=O)cnc(S)nc1 Cc1c(C(=O)NC(C)(C)CC(=O)N2CCC(N3CCC3)CC2)cccc1O c1(OCC)ccc(C)cc1C(CCN)N1CCCC1.N12N(CCC1=O)C2=O.SC C1(NC(C(CC)NC(C)=O)=O)CCC12CN(C(c1ccnc(C)c1N)=O)C2 c1(C(C(=O)N(CCN(C(C)C)C(C2CCN(C)C2)=O)C)(C)C)c(F)cccc1F C(=O)(C(C)(C)CCNC(=O)C(N1CCOC1=O)C)NCCc1c(C)nccn1 C(C)(C)(CC(=O)NCC(CC(C)C)NC(=O)C(F)CC1CCC1)OC N1(C(c2cc(C)c(O)cc2)=O)CCC(C)(C)C(C(N2CCCC2CC(N)=O)=O)C1 c1(C(N2CCC(NC(C3CC(C)C3)=O)C2)=O)cc(C)n(-c2ccc(F)cc2)n1 N1(C(CCCN(C(C)=O)C)=O)CCCC(N(C)C(c2ncnc(C)c2C)=O)CC1 c1(C(=O)NCC2CN(C(C3(F)CC=CCC3)=O)CCO2)cc2cccnc2s1 C1(NC)CCC(N=c2cc[nH]cc2S(=O)(=O)NC(N2CCC(N)CC2)=O)CC1.OC c1(NC(C(c2cn(C)nn2)NC(CCC#C)=O)=O)ccc2c(c1)CCO2 N1(C(C2(C#C)CCCC2)=O)CCN(C(C2CCC2=C)=O)CC1C C#Cc1cc(C(=O)N(CC(=O)N(c2cccc(C)c2C)C)C)ccc1C N1(C(CCC2(C)N=N2)=O)CC2(CCCC2NC(=O)CC2CCCS(=O)(=O)C2)C1 N1(C(CC(=O)OCC)=O)CCC2(CC2NC(=O)CCOCCOC)C1 C1(CCNC(C(=O)NCCOC)=O)CCN(C(=O)CC2CNC(=O)C2)C1 CCCCCCCCC(=O)NCC(C(=O)NCC1(C2CC2)CCCO1)C(C)C c1(C(=O)NCC(C)(C2CC2)NC(C2CC(C)SCC2)=O)nc2c(s1)CCCC2 N1(C(CCC(C)OC)=O)CC(CNC(c2ncc(N(C)C)cn2)=O)CC(C)(C)C1 C=C1CCCN(C(=O)C(CN(C)C)NC(=O)Cc2ccoc2)C1 c1(N2CC3CC(CN(C(CS(CC)=O)=O)C3)C2)ccc(OC)c(F)c1[N+](=O)[O-] c1(OC)ccc(C(=O)NCC(C)NC(=O)Cc2cc[nH]n2)cc1S(N)(=O)=O c1(CC(=O)NCCN(CCC)C(c2cccc(=S)n2O)=O)cc(O)nc(O)n1 C=CC1(CNC(C2OCCC2C)=O)CCN(C(=O)C=CC2CCC2)CC1 C1(NC(C(C)OCCN(C)C)=O)C2CC3C1C3C2C(N1CCC2CC12C)=O N1(C(=O)Nc2nn(-c3cccc(Cl)c3)cc2O)CC(C(F)(F)F)CC1=O C=C(C)CC(C(=O)NOCC1(C)CC1)NC(=O)CC1CCCCCC1 CCC(CNC(=O)C(CCSC)NC(c1cnsc1C)=O)(CC)CO c1(COC)nc(C(=O)NC(C)CNC(C2CC2(Cl)Cl)=O)co1 C(CNC(c1coc(C(F)F)n1)=O)(C(C)(C)C)NC(c1c(C(C)C)c[nH]n1)=O N12C(=O)NC(C(C(=O)N=c3cc(C(C)(C)C)o[nH]3)C1F)C2(C)C.CCOC CC(CC(=O)NCC1CC2CN(C(c3cccc(C(N)=O)c3)=O)CC12)C(F)F N1(C(c2ccc(C)c(C(F)(F)F)c2)=O)CCC2CCC(NC(=O)CC(C)CF)C12 c1(COC)nc(=NC23CCCC2CN(C(=O)CC2CC4(CCOCC4)CO2)C3)s[nH]1 C(CCS(C)(=O)=O)(C(=O)N1CCC(O)(CCNC(=O)C(F)=C2CCC2)C1)OC N1(C(Cc2c(C)nsc2)=O)CCCC12CCN(C(C1(CO)CCC1)=O)C2 C1(CCNC(N(C2CSC2)C)=O)CCCNC1=O Cc1c(C(=O)NC2CN(C(C3CC3[N+](=O)[O-])=O)C2)cccc1N1CCNC1=O c1(C(N2CC(C)(NC(c3n(CC)ccc3)=O)C2)=O)[nH]c(=N)sc1-c1ccccc1 C(=O)(CC(C)(C)C1CC1)N1C(C(N(C2CC(=C)C2)C)=O)C=CC1 c1(CC)nc(C(N2CCC(N(C(C3CC(CCO)C3)=O)CC)C2)=O)cs1 O=C(CCC(CF)CF)NCCSCC(N1CC2=NC(CC2)C1)=O C12(CNC(CNC(C)=O)=O)CCC(C1)N(C(c1c(C)noc1C(F)F)=O)C2 Cc1nnsc1C(C)NC(=O)C(C1CC1)N(C(=O)Cn1cccc1)C N1(C(C(C2CCCOC2)OC)=O)CCN(C(=O)CCc2nncs2)CC12CCC2 c1(OC)cnc(C(=O)N(CCNC(=O)COC(F)F)CCOCCO)cn1 Cn1cc(-c2ccoc2C(=O)NCC(CO)NC(=O)CNC=O)cn1 Cc1c(Br)c(C(=O)NCC2(C)CCCN2C(C2C(C)C2C)=O)nn1C C#CCCCC(C)C(=O)N1CCC(NC(=O)CCc2cccc(Cl)c2Cl)CC1C N1(C(CC(C)F)=O)CC2(NC(=O)COc3ccc(Cl)nc3)CCC1CC2 C(CS(=O)(=O)C1CC1)N(C(=O)NCC(n1cccn1)C)C C1(CC)CN(C(=O)CCC(C)(C)C)CCC1NC(c1nc(C2CC2)cs1)=O C(C)(CCCCNC(C1CCC(F)CC1)=O)NC(c1c(CC)nc[nH]1)=O C1(CN2CCC(N(C3CCN(C(=O)OCC)C3)C)C2)CCOCC1(C)C N1(C(CCCOCCC)=O)CCC2(CCN(C(C3(CCO)OCCO3)=O)C2)C1 C(=O)(C1CCCc2sccc21)NC(CNC(C(C(C)O)NC(N)=O)=O)C(C)(C)C c1(C(N2CC=CC(NC(Cn3nnc(C)n3)=O)C2)=O)ccc(=O)n(C)c1 CCC(C)C(O)C(=O)NCC(C1CCCCCC1)NC(c1ccc(C(N)=O)[nH]1)=O N1(C(CC(CC)N(C)C(c2ccc(=N)[nH]c2)=O)=O)CCN(C)CC1CO c1(OC)ncnc(C)c1C(=O)NCC(CNC(=O)CC1CCCCO1)S(C)(=O)=O C1(CC(=O)NCC(Cc2ccccc2)C(=O)O)COCCOC1 c1(C(=O)NCCC2CCCN(C(CC=C=C)=O)C2)ccc(O)cc1CC CC(C)CCCCC(=O)N1CC(OCCC(N2CCC(SC(F)F)C2)=O)C1 N#Cc1cccc(NCC(N2CC3CC(NC(c4coc(Cl)n4)=O)C3C2)=O)c1 CC1OC2(CO)CC1(C(N1CCCC(NC(c3ccn(C)c3)=O)C1C)=O)C2 C1(CNC(CSCC(C)C)=O)CCCN(C(C2CCC(O)CC2)=O)CC1 c1(CC(=O)NC(CC)(C)CNC(c2cnc(C(C)=O)s2)=O)cccc(OC)c1 Cn1cc2c(n1)CCCC2C(=O)N1CCC2(CCCN2C(c2cnns2)=O)CC1 C1(C(=O)NCC(C)(CO)NC(c2ncc(NC)nc2)=O)CCn2cnnc2C1 CC(C(=O)N1CCC(O)(CNC(=O)C(O)Cc2cnc[nH]2)C1)S(C)(=O)=O C1(CC=C)(C(=O)NCC2(CC3CC3)CCC2)CN(C(=O)C=C(C)C(C)C)C1 C#CC1(C(N2CCC(CCC(=O)NC(C)C(C)SC)C2)=O)CC(=O)C1 C1(C(=O)OC)CN(C(c2n[nH]c(=N)s2)=O)CC1N c12cccc(c1)C(=O)NC(C)CNC2=O.c1(Cn2cccn2)ncsc1C1CC1 c1(OC(C(N2C(CC)CCCC2)=O)NC(C23CCC(C2)C3)=O)c(C)cccc1Br C=C(C)CC(C(=O)N1C(C)CCC1(C)C)NC(c1cccc(CC)n1)=O C1(C(=O)NCC23OCC(CNC(C4CCCSC4)=O)(C2)C3)CCC2CC1CO2 CC(O)C(F)(F)C(=O)NCCN1CCN(C(C2(CN(C)C)CC2)=O)CC1 C(=O)(C#CC1CCOC1)N1CC(C(=O)NCc2cnn[nH]2)OCC1 CCCC(C)(CCC)C(=O)NCC1(CNC(=O)C2CCc3nccn32)CC1 N1(C(C2CC(CCC)OCC2)=O)CC2CC(C1)C2NC(=O)CC1CCCCC1 CC(C)CC(C(=O)N1CC(CNC(C2(S(C)(=O)=O)CC2)=O)C(F)(F)C1)N(C)C C#Cc1cccc(C(N2CCCCC2CCNC(=O)CSCC=C)=O)c1F N1(C(C2CC(CCC)C2)=O)CCC(NC(=O)C=CSC)C(CO)C1 Cc1ccsc1CC(=O)NCC1CCC(C(N2C(CN(C)C)CC2CO)=O)O1 c1(OCCC)cccc(-c2ccc(NC(C3CC3F)=O)cn2)c1F c1(C(=O)Nc2cc(C)cc3c2nccc3)coc(C2=CCC(C)CC2)n1 Cc1cc2[nH]c(C(=O)NCC3CCCN(C(C4CC(C)(O)C4)=O)C3)cc2s1 C(=O)(C1=C(Cl)CCC1)NC(CCNC(C(F)=CCC)=O)(C)CC c1(N(C)C)nc(Cl)c(C(N2CCOC(CNC(C3CCCCO3)=O)C2)=O)s1 C1(CC(=O)Nc2ccsc2)CCCC1(F)F.C12(CCCC1)CCNC(=O)COC2 c1(OC)ccc(OC)c(OC)c1CCC(N1CCC(CO)C(O)CC1)=O CN1CC2C(C(=O)NC(C(=O)NCC(=O)N3CCCO3)C3CCOC3)C2C1 C1(CNC(c2c(CCC)nco2)=O)CC2(CCC2)CN1C(=O)COCCCOC c1(C(=O)NC2CC(CNC(C3C(SC)CCC3)=O)C2)ccc2n[nH]cc2c1Cl C(=O)(CCC(C)(C)C)NCCCCNC(CCCCSC)=O C=CCC(CNC(=O)CC(C)C(C)C)C(=O)NCCCn1ccnn1 C1(C(=O)NS(C(c2ccccc2Br)C)(=O)=O)C(C2CC2)C1(F)F C1(CO)CCCCC1.C1(CCC)CC1C(=O)NCCNC(=O)C=CCOC Cc1nc2ncnn2c(NC(C(C)NC(=O)CCC2(C)CC2)C(C)C)c1C c1(C(N2CC(CCNC(COc3cn(C)nc3)=O)OCC2)=O)csc2nccn12 CC(C)CCC(C(=O)O)NC(=O)Nc1cccc(C2CNC(=O)C2)c1 C1(CNC(CC=C)=O)CN(C(c2ccn(CC)c2C)=O)C2CCCC2O1 C1(N(C)C(C2CC=CC2)=O)CN(C(=O)C(N)=O)CC1(C)C N1(C(C(CC(=C)C)OC)=O)CCC2CCN(C(=O)C(C)C3(O)CCC3)CC12 N1(CCC(=O)N(CCN(C(C2CCC(C(N)=O)C2)=O)CC)CC)CCCCC1 CC(C)(C)C#CC(=O)NCC1(O)CN(C(C2(N(C)C)CCCSC2)=O)C1 N1(CC(N2CCCC(CN(C)C(C3(C)CCCN3C)=O)C2)=O)CCCOC1=O CC1CCCC(C)C1NCC1CC2(CC(=O)N2)C1 CCCCCCCC(C)CNCc1cc(-c2c(F)cccc2F)on1 c1(CNC2OCCC(Oc3ccc(COC)cc3)C2)nc2ccccn2c1Br C(C(F)(C(=O)NCC1(C)CCCC(=O)N1)C(C)C)NC(C=C(C)C)=O c1(CC)ccc2c(c1)C(=O)C(=O)N2.c12nc(cc(C)n1)NC(=O)CS2 c1(C(=O)NCCCN(CCC)Cc2ccccc2)nnc(COC)o1 c1(CN2CC3C(NS(CCCC)(=O)=O)(C3)C2)c(N)ccc(C(=O)OC)c1F C1(CC(=O)NCC(CC(C)C)(C)O)CN(C(=O)CC2CCOC2)C2(CCC2)C1 C1(COCCOC)=CC=C(S(=O)(=O)NNS(=O)(=O)c2ccc(S(C)(=O)=O)cc2)C1 C1(CNC(C(C)CC2CCCC2)=O)CC2(CC2)CN1C(=O)C1=NOC(C)C1 C(CC(C)C)(C(=O)N1CCN(C(C2CCSCC2)=O)C(CF)C1)NC(C)=O N1(CC(=O)NCc2ccc(Br)cc2)CC(F)(F)C(F)(F)C1 C=C=CCCCN=C(NCc1ccnn1C)NCC1CCCC(C(C)C)C1 c1(C(=O)NCC#CCNC(C(CC=C)NC(C)=O)=O)ccccc1N=NN(C)C c1(OCCC)ccc(N2CCCC2COC(c2nnnn2CCC(F)(F)F)=O)cc1 C12(C(N(CCNC(CC(CC)CC)=O)CC3CC3)=O)CCCCC1CS(=O)(=O)C2 C1(C(=O)NCCC2C(CC)C2)CC(O)(CNC(=O)CCn2cc(C)cn2)C1 C(CC(C)C)(C(=O)NOCCC(F)(F)F)NC(C1CC(C)(CC)C1)=O CC1(C)CC(NC(c2cc3occc3[nH]2)=O)CN1C(C1CC2C=CC1C2)=O c1(C(=O)NCCC2CN(C(C(C)(C)C3CCOC3)=O)C2)scc2c1OCCO2 n1(CC(=O)NCCCCNC(C2CCOC2)=O)cccnc1=O Cc1ccc2[nH]c(C(=O)NCC3CC3CNC(=O)CNCC3CC3C)cc2c1.SCC Cc1ccc(C(=O)NC23CCCN(C(=O)C=C4CCN(C)C4)C2C3)c(=O)n1C N1(C(CC(C2CC2)NC(CCOCCC)=O)=O)CC23CCC2(COC3)C1 C12(C(=O)NCC3CC(CC)C3)C(NC(c3ccc(NC)cc3)=O)C3CC1C2C3 c1(NC(=O)OC)ccc(S(=O)(=O)Nc2nccc3cc(C#N)ccc23)c(Cl)c1 Cc1ccc(O)c(NC(C2(CCNC(=O)C(F)C(C)(C)O)CCCC2)=O)c1 c1(C(=O)NC2(CNC(c3cnc(C)[nH]3)=O)CCCCC2C)cccc2nc[nH]c12 CC(C)CN=C(NC1CC1C)NC1CCC(O)C1.c1(C)ccc(F)cc1 C1(CNC(C2CC2C(F)F)=O)CC12CCN(C(c1ccnn1C(F)F)=O)CC2 c1(OC)ccc(OC)c(C(N2CCN(C(C3CC4CC4C3)=O)C(C(F)F)C2)=O)c1 C(C1c2ccccc2CCN1C(=O)Cn1cnc(C#N)n1)NC(C(CC)CO)=O c1(C(=O)NC(C(C)C)C(C)NC(c2cscc2Cl)=O)cc(N)cc2c1OCCO2 CC(C#N)CN=c1[nH]c2c(c(=NCC3CCCCS3(=O)=O)[nH]1)CCC2 n1(CCSC)nnnc1C(C1(C)COC1)NC(C)Cc1ccnn1C N1(C(c2c(C)ccnc2)=O)CCC2CCC(C1)N2C(=O)Cn1cnnc1 Cc1oc(CNC(=O)C(N2CCNC2=O)C)nc1C(=O)NC1CC1F CC(C)(C)CCCC(=O)NC1CC2(C1)CC2C(N1CCCC(CCF)C1)=O S(=O)(=O)(c1cccs1)NCC(=O)NCC1(CN(C(CC=C)=O)C)CC1 C1(C(=O)NC(C2CCCN(C(c3nccn3C)=O)C2)C)CSCC(=O)N1 c1(C(ON(C(=O)c2ccc(C(C)O)cc2)C(C)C)=O)cc(F)cc([N+](=O)[O-])c1.CO S(=O)(=O)(c1csc(C(F)(F)F)c1)N1CCN(CCCNC(C(C)N(C)C)=O)CC1 Cc1n[nH]c(C)c1CCC(=O)NC1CC1CNC(c1csc(CC(F)F)n1)=O CC1OC2(CNC(=O)C3CC3)CC1(NC(=O)CCc1cc(F)ccc1Br)C2 C(=O)(C1=NOC(C)(C)C1)N1C(C(C)NC(c2ncn3c2CCC3)=O)CCCC1 c1(C(N2CC3C(CNC(c4scc(C)c4)=O)C3C2)=O)cc(C(C)C)ccc1N C(=O)(C(F)(CNC(c1sc(O)nc1C)=O)C(C)C)NCC(COCC)O N1(C(C2(OCC)CCCC2)=O)CCC2CCC(NC(c3cc(C#N)c[nH]3)=O)C1C2 n1(CC)cnc2nc(=NCCC3CC3)[nH]c(NCC3(CS(C)(=O)=O)CCC3)c12 CCCC(C(=O)NC(CN(C(=O)Cc1ccccc1C)C)CC)C(C)C C#Cc1ccc(C(N2CCC(c3nncs3)CC2)C(=O)NC2CCCCC2)cc1 N1(C(CCc2n(C)cnn2)=O)CCN(C(c2ncncc2N)=O)CC(O)C1 C1(OC)CCCC1C(=O)NCC1CC1CNC(=O)Cn1nnc(C(C)(C)C)n1 Cc1ccc(C(=O)NC2COCCC2NC(C23CC(C)(CO2)C3)=O)n1C C1(CNC(C=CC(C)(C)C)=O)(CNC(C2CCN2C2CCCC2)=O)CCCC1 C1(NC(c2cnc(O)s2)=O)CC12CCN(C(=O)C(F)(F)C1(O)CCC1)CC2 c1(OC)cncc(C(=O)N(CC(C)N(C)Cc2nc(N(C)C)n[nH]2)C)n1 C(=O)(C(C)(C)CS(N)(=O)=O)N(C)CC1COCCN1C(=O)CC1CCCO1 C(=O)(CCCCC(=O)N1CC2CCC1C(CNC(C13CC(C1)C3)=O)C2)OC C1(CCC=C)(C(N2CC(C(=O)OC)C2)=O)CN(C(c2ccncc2)=O)C1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1CCCC(NC(C2(C#N)CC2)=O)C1 CC1CC(NC(=O)CCCCN2CCOC2=O)CN(C(C2CC=CCO2)=O)C1 C1(C(N)=O)CCCC(CNC(C2CC(O)(CNC(c3n[nH]cc3Cl)=O)C2)=O)C1 c1(C(=O)NCCc2cc(C(=O)NCCc3cncc(C)n3)no2)c(C)ccnc1O CC1CCN(C(c2ncoc2Br)=O)CCN1C(c1ccn(CCF)n1)=O CC1OC(=O)NC1C(=O)NCC1CN(C(c2cc(O)ncn2)=O)C1 C(=O)(C(C)(C)CS(C)(=O)=O)NCC1CCN(C(c2c(C)onc2CO)=O)CC1C C1(C(=O)NCC2CN(C(C3CCC3(C)C)=O)C2)(COC)CCC(=O)N1 Cc1nc2n(n1)CC(C(N1CC(CNC(C34CC(CO3)C4)=O)OC(C)(C)C1)=O)CC2 C(=O)(C(CCOC)NC(=O)C(C)Cn1ccnc1)NCCc1n(CC)cnn1 c1(C(=O)NCC2(O)CCN(C(COC(C)(C)C)=O)C2)ncnc2c1CCC2 N1(C(C2CC2C(F)F)=O)CCN(C(c2cn(C3CCC3)nn2)=O)C(C2CC2)C1 CC1COCCN1CC(N1CCC1CC(=O)NCCc1cccc(F)c1)=O c1(N(C(C(n2cc(C(CSCC)C)nn2)(F)F)=O)CC)cnc2c(c1)COC2 N1(C(c2ccc(OC)cc2C)=O)CC2CCC1CN2C(C1CC1(C)C)=O C1(NC(CCc2n(C)cnn2)=O)CCCCCC1C(N1CC(S(C)=O)C1)=O Cc1ccc(C(=O)NCC)cc1NC(=O)C(C)(C)C.C1(C=O)COCC(C)(C)O1 CC(C)(C)C(CNC(c1ccc(F)c(O)c1)=O)C(=O)N1CCCCC1CCCO C1(C(=O)NC2CCCN(C(c3c(C)cnn3C)=O)C2)CCCN(S(N)(=O)=O)C1 C1(C(N2CC(O)(CNC(C3CCCC3(F)F)=O)C2)=O)CCC2C(C1)C2(F)F N1(C(CN(CCCC)C)=O)CCCC(Cn2cc(COC3CC(F)(F)C3)nn2)C1 C=CCCC(C)(C)C(=O)NCC1CC(F)(CNC(c2nocc2C(C)(C)C)=O)C1 C1(CNC(CSCCC)=O)CC2CCC(C1)N2C(c1cnc(C(C)C)[nH]1)=O CCC(C)(C)C(=O)NCc1cn(CC2CC(C)N(C(c3ccc(F)cc3)=O)C2)nn1 C(=O)(C1=CCc2ccccc21)NC1C(NC(=O)CCCCC(F)(F)F)CCCC1 c1(C(N2CC(C(=O)OC)OCC2)C(=O)NCCCF)c(C)cc(C)n(C)c1=O c1(OC)noc(C)c1C(=O)NCC(C)N(C)C(C1(Oc2ccccc2)CC1)=O C(=O)(CC(C)CC(=O)N1CCC(NC(=O)C2CC2)CC1C)OC CC1(C)CCCC(C(N2CC(C(F)Cn3cc(C4CCCCC4)nn3)C2)=O)CC1 c1(C(N2C(C)CCC(NC(C3CCCCN3C)=O)C2)=O)cccn2ncnc12 Cc1nc(OC(F)F)c2sccc2n1.c12ncccc1N2.C12(C)CCN1C2=O CC1(C)CCC(F)(F)CC1C(=O)NC1CCC1NC(=O)CN=S(C)(C)=O C1(C(=O)OC)CCC2(CC1)CC(NC(=O)Nc1ccc(C(=O)N(C)C)cc1)C2 C(CC(C)C)(C(=O)N1CC2CC2C1C(N1CCC(C)(N(C)C2CC2)C1)=O)OC c1(C(=O)NC(C(=O)NC(c2nnnn2C)C)(C)C)cc(C#N)n(C)n1 C1(NC(Cc2c(C)noc2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1F O=CN1CCCC1C(=O)NCCC1CCN(C(C2(c3ccno3)CCC2)=O)CC1 c1(OC)ccc(C(N2CCN(C(=O)CCC3CC(OC)C3)CC2C)=O)c(Cl)n1 C=CCC(C(=O)NCCc1nc(C)oc1C)NC(=O)CCN1CCCC1=O C(=O)(C1CCC(=O)c2cccn21)NC1CC(NC(c2nc(C(C)(C)C)oc2)=O)C1 C(CCCC)(CC(=O)O)NC(CC(CC#C)c1ccccc1)=O N1(C(C(CC)(CC)CO)=O)CCOC2(CCCN(C(=O)CCCOC(C)=O)C2)C1 Cc1c(C(=O)N(C)CCNC(=O)CC2CC3CCC2C3)oc(=O)c2ccccc12 c1(C(N2CCC(N(C)C(c3cccs3)=O)C2)=O)c(Br)ccc2n[nH]cc12 CCC(C)CCCC(=O)N(CC(C)NC(c1ccnc2c1CCC2)=O)CC C(C(C)C(=O)NC1CCCC1O)N(C(C=CCC)=O)C c1(C(N2C(CNC(C3(SC)CCC3)=O)CCC2)=O)cccc(N)c1Br c1(CC)noc(CN2CCCC2C(=O)NCCCCN2CCCC2)n1 C(=O)(C(C)(C)C(F)(F)CC)NCC(CCCC)NC(c1cn2cccnc2n1)=O CP(C)(=O)c1ccc(C(N2CC3CCC3(CNC(c3cc(CO)on3)=O)C2)=O)nc1 CC(C)(C#N)CCCC(=O)NC1(C2CN(C(C3CC4CC4C3)=O)C2)CC1 C12(NC(C3CC(OC)C3(C)C)=O)CCC(CC1)N(C(=O)CCCC(C)C)C2 c1(C(=O)NC(C)CCNC(c2ccc(Cl)c(F)c2O)=O)cc2ncn(C)c2cn1 C1(CN(C(=O)C(c2ccc(Cl)cc2)O)C)CCCN(C(c2cnn[nH]2)=O)C1 C1(CNC(c2ccc(C)cn2)=O)CC2(CC2)CN1C(c1cc(N)ccn1)=O C1(C(=O)NCC2(F)CN(C(c3c(CC)[nH]c(=N)s3)=O)C2)CNC(=O)CC1(C)C C(=O)(C(F)C(C)CNC(c1c[nH]nc1Cl)=O)N(C(C)C)CC N1(C(C2CCC(CC)O2)=O)CCCC(C)(CNC(=O)CC2(OC)CCOCC2)C1 C1(C(=O)NCc2ccc(F)nc2)CC12CCN(Cc1c(F)cc(Br)cc1F)CC2 C1(C(N(CCCC(F)(F)F)C)=O)CC2(CCN1C(=O)CC1NC(=O)NC1=O)CC2 O=C1CN(Cc2noc(C3CC3)n2)CCN1.C1(=O)C(=O)NCC2C(C2)N1 CCCC(C(O)C(=O)NC1CCOCC1C)NC(C1CC2(CCO1)CC2)=O CC(O)C(F)(F)C(=O)N1CC(NC(c2cc(Cn3cccn3)on2)=O)CC(F)C1 C1(C(=O)NCCC2CCN(C(Cc3[nH]c(=N)sc3)=O)CC2)CCOCC12CCC2 c1(-n2c(C(CCCCCC#C)NC3(C)CCC3)nnn2)ccc2c(c1)OCCO2 Cc1cc(OCC(=O)NCC2C(C)CCCN2C(c2cscn2)=O)cc(C)c1 c1(OC)cccc(O)c1C(=O)NCC1CCN(C(=O)C(C)S(C)(=O)=O)C1(C)C C(N=c1[nH]c(=NCC2CCCOC2)[nH]c2c1COC2)c1snc(C(C)(C)C)n1 C1(C(=O)NC2(C)CCN(C(CCCC)=O)C2)CCC(C2CCC2)CC1 c1(OC)c(C(=O)NCC2(O)CCN(C(c3cnc(C)cn3)=O)CC2)c(C)nn1C CCCCCCCCC(=O)Nc1cncc(-c2cccc3c[nH]nc23)c1 c1(OC)ncc(C(=O)NCCC(O)CNC(C2(C)CCCS2)=O)cc1C N1(C(C2C(CCC)C2)=O)CCC(O)(CNC(C2COCCN2CC2CCC2)=O)C1 Cn1nnc(Cl)c1C(=O)NCCC1CC(NC(=O)C=CCO)C1 C1(OC)C(NC(=O)C(C)(C)NC(=O)CC2CCC3CC23)CC1O C1(CNC(COCC=C)=O)C2CC1N(C(c1ccncn1)=O)C2 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)NCCN(C)C(C12CC(C)(C1)OC2C)=O C1(NC(C2C3CN(C(CC4C(C)(C)CCO4)=O)CC32)=O)CCCC2CCCN12 N1(C(c2cn(CCCC)nc2C)=O)CCC(C)N(c2nc3ccccc3s2)CC1 c1(OC)cc(OC)c(C(N2CCC(O)(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)c(N)c1 c1(CC2N(C(=O)CC3(O)CCSC3)CCCC2)ccc(F)c(F)c1 C1(C(N2CCN(C(C(F)=CC)=O)C(c3ccncc3)C2)=O)CC(C)CC(C)(C)C1 CC(C)C(C(=O)N1CCCCC1CCO)NC(=O)C(F)F c1(C(=O)NC23CN(C(CC(C(=C)C)OC)=O)C(CC2)C3)cccn2nncc12 Cc1c(C(=O)NCC(C)NC(=O)CC2CCC(O)C2)cccc1C#N N1(C(c2c(C)cccc2)=O)CCCC(NC(=O)COc2cccc(F)c2)C1C CC(C)(CC#N)C(=O)NCCCOCCC(=O)NC1CCCCCC1O C(=O)(C1COc2ccc(Br)cc21)NC1CCN(C(C2(CC#C)CC2)=O)C1 C(=O)(C1=CCC(C)CC1)NC1CCN(C(c2cncc(C)c2)=O)C1 C(=O)(C(C#N)C(C)(C)C)N(CCOC)CC1CC1.C12(CCCO1)C(=O)NC2 N1(C(C2C=CC(NC(C3C(COC)CC3)=O)C2)=O)CC(N=[N+]=[N-])C1 N1(C(C(COC)O)=O)CC(C)OC2(CCN(C(c3cccc(C)c3Cl)=O)CC2)C1 N1(C(CC(C)=C(C)C)=O)CCC(C(=O)N(C)CC2(O)CCC2)C1(C)C c1(C(=O)NC2N(c3nc(C)c(Br)cn3)CCC2O)cc2ccccn2n1 C1(CC(=O)N(C2CN(CC3CCCCC3)C2)CC2(O)CCSC2)CC2(CC2)C1 O=C(C1CCCc2ncccc21)NC1CCN(C(c2cccc3ccccc23)=O)C1 Cc1cc(S(N)(=O)=O)oc1C(N1CCCC(N(C(=O)COC(C)C)C)CC1)=O N1(C(C2(F)CN(C(C3N(CC)CCCC3)=O)C2)=O)CC2CCCN2CC1C c1(CC(N2CCCC(N(C(=O)CCc3ccc[nH]3)C)C2)=O)cc(O)nc(O)n1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(CCNC(C(CCSC)O)=O)C1 C(C(F)(C(=O)NCCCC1CCOC1)C(C)C)NC(c1c(C)noc1C)=O c1(C(CCC)NC(=O)C(C)N(C2CC2)CC)cn(-c2nccs2)nn1 C1(CCC(=O)NCCN(CC(F)F)C2CC2)CC2(CCC2)CCO1 N1(C(c2ccc(F)c(C)c2N)=O)CCC2CN(C(=O)Cn3ncn(C)c3=O)CC12 CCCC(C)(C)CC(=O)N1CCC(NC(c2cn(C)cn2)=O)CC1C c1(CCC(=O)N(C2CN(C(=O)C=Cc3ccc(Cl)s3)C2)C)cc(F)cc(F)c1 C1(C2(N(CC(N3CCCCC3CCCO)=O)C3CC3)CC2)COc2ccccc2O1 C1(C(=O)NC2(CN(C(c3cccc(CC=C)c3)=O)C)CC2)COCC2(CCC2)O1 Cn1cc2c(C(N3CCCC4CN(C(=O)C5=CCCSC5)CC34)=O)cccc2n1 N1(C(CNCc2cn(C)nc2)=O)CC2CC1(CS)C2.c1(C2C(O)C2)ccc(Cl)cc1 N1(C(C(C)CO)=O)CCC(c2cccc(F)c2)(NC(c2cc(CN)ncn2)=O)C1 c1(C(N2CCC(C)(CCNC(C3CCC(F)(F)C3)=O)C2)=O)ccc(C#N)c(Cl)c1 C(C(=O)N(CC(=O)NC(COCC)CC)C1CC1)(C(C)C)OCC C(=O)(CS(=O)(=O)NC(C)(C)C)N(C1CN(C(c2csc(-c3cnc[nH]3)n2)=O)C1)C N1(C(CCC(C)OCC)=O)CCC2(CC2C(=O)NCC2OC(=O)NC2(C)C)C1 C1(NC(C=CC2(C)COC2)=O)CCN(C(=O)CCCCn2ccnn2)CCC1CO CC1CC(NC(c2cnco2)=O)CCN1C(=O)C(F)C(C)(C)O C(CN=c1ccc(S(=O)(=O)NCc2c(F)cccc2F)c[nH]1)c1scc(CC)n1 c1(C(CC)(C)C)ccc(CNC(c2nnnn2C(C)C)(C)CSCCC)cc1 C1(NC(CC(C(=C)C)OCC)=O)CC2CC1CN(C(c1ccc(C)c(C)c1)=O)C2 N1(C(c2c(O)ncc(CC)c2)=O)CCC(C)N(C(C2CCCCS2(=O)=O)=O)CC1 C1(NC(C(CC)F)=O)CCCC2CN(C(c3cc(C(C)C)n(C)n3)=O)CC12 c1(SC)cc(C(=O)NC(C2(O)CN(C(=O)C(C)(C)c3ccccn3)C2)C)co1 c1(C(=O)NC(c2ccc(CNC(C(C=CC)O)=O)cc2)C)cc(=N)[nH]c(Cl)n1 C1(CNC(=O)Cn2cnnc2O)CC2CCC1N(C(C1C3CCC(=O)C13)=O)C2 Cc1ccc2cc(CN(C=O)Cc3ccc(-n4cccn4)cc3)ccc2n1 c1(NC(C2N(C(C3(C(=O)OCC)CC3)=O)C(C)C2)=O)ccnc2cc(Cl)ccc12 c1(C(N(C2CCN(C(c3c(C#N)ccs3)=O)C2)CCO)=O)c(F)ccc(O)c1F C1(NC(CC(C)F)=O)CC2(CCC(CNC(=O)CCCN(C)C)CC2)C1 N1(C(C2CN(C(C(C)S(N)(=O)=O)=O)CC2(F)F)=O)CC2(CCN(C)CC2)C1 n1(CC(C)C)nc(Cc2ccsc2)nc1-c1ccc(-c2cccs2)o1 Cc1c(F)cccc1S(=O)(=O)N1CCC(N(C)C(c2c(F)cc(F)cc2Br)=O)C1 C(=O)(CCC(F)(F)F)NC(CC(C)NC(c1csc(-c2ccc(F)cc2)n1)=O)C c1(NC(CC(C)OCc2ccccc2)=O)nccc(=NCCC2=CCOCC2)[nH]1 c1(OC)ccc(Cl)c(CNC(=NCCF)NC(C)CC2CCCO2)c1 c1(OC)ccc(Cl)nc1C(=O)N(C1CC(NC(=O)C(=O)N(C)C)C1)C C(CCNC(=O)C(=O)Nc1ccc(Cl)cc1)(C(C)C)NC(C(CC)C)=O c1(C(=O)NCC23N(C(C(=O)c4ccco4)=O)CCC2CC3)c(F)ccc(Cl)c1F Cc1ccc2ccc(C(N3CCN(CC4CCCC4)CC3C)=O)nc2c1 N1(C(c2cc(CNC(C3C(C)C3)=O)ncc2)=O)CCC2(C1)CC2(F)F c1(C(N2CC3CCN(C(c4cnc(C)[nH]4)=O)C3C2)=O)c(O)nnc2c1CCC2 c1(NC)ccc(C(=O)NC2CCCCC2NC(C23CC(OC)C2C3)=O)nc1 c1(CCN(C(CCNC(C)=O)=O)CC)ccn(C)n1.C(=O)(C=CC(=O)N(C)C)N N1(C(C2CCCN(N(C)C)C2)=O)CC2CC1CN2Cc1cc2n(n1)CCC2.C=O C1(NC(CCCC)=O)CN(C(c2cncn2-c2cnn(C)c2)=O)CC1O C(=O)(CCC(=O)NCCCC(C)NC(C1CC2CCCC12)=O)NCCC C1(O)(CNC(CN(C(C)=O)C)=O)CCN(C(C2(CC(C)=O)CCCC2)=O)C1 c1(OC(C)C(=O)NCCNC(C2COC(=O)N2)=O)ccc(Cl)cc1Cl c1(C(=O)NC2CCCCC2C(=O)NCc2cscn2)c(F)cccc1Cl Nc1c(-c2ccccc2)nsc1C(N1CCC(CNC(C23CC2CC3)=O)CC1)=O C1(NC(c2coc(C(C)C)n2)=O)CCOCC1C(=O)NCC1CC2(CCC2)C1 N1(C(C(C)(N(C(=O)CC2CC(C)(C)CO2)C)C2CC2)=O)CCCC2C1CCN2C CC1(C)CCOC1CC(N1CCCC1C(N1CC(n2ccnn2)C(O)C1)=O)=O C1(NC(c2cn(C)nc2)CC2CC2)CCC2(CCCC2)C1 c1(C(=O)NCCOCC)ccc(C(C(=O)OC(C)(C)C)C(C)C)cc1.C(CC(=O)OC)=C N1(C(C2C(C)CC2)=O)CCC(C(C)(C)C(=O)N(CCc2ccccc2)C2CC2)C1 c1(C(C(=O)N(CCNC(C(C)NC(=O)NC)=O)C2CC2)O)cccc2ccccc12 CCCCC(O)C(C)C(=O)NC1CN(C(=O)Cc2cc(F)ccc2F)CC1CC CCCCC(O)CC(=O)N1CC(CCCCNC(c2cnn(C3CC3)c2C)=O)C1 c1(C(n2cc(C(C)NC(=O)C(c3cccnc3)C)nn2)C)cccc(F)c1 C#CC1(NC(=O)CC2CC(NC(C3CC(N4CCCC4)C3)=O)C2)CC(F)(F)C1 c1(CCC(=O)NCCNC(C2CC3CC2C3)=O)ccc(C2CC2)cc1 CCC(CC)CC(=O)N1CCC(NC(c2ccnnc2O)=O)CC1C1CC1 c1(C(N2CC(NC(COCC=C)=O)CC(F)(F)C2)=O)cccc2c(C)c[nH]c12 C(CNC(=O)Cn1cnnc1O)(CC(F)(F)F)NC(c1ccc(CCC)cc1)=O c1(C(N2CCC(CC)C2C(=O)NCCCc2cnccn2)=O)cc2n(n1)CCO2 CN1C2CCCC1CN(C(C13CC1CCN3C(C1CC1Cl)=O)=O)C2 Cc1cc(C(=O)N(C2CCN(C(=O)CC3(C)CCC3)C2)C)n(C2CC2)n1 N1(C(CCc2ccc(C)nc2)=O)CC(C(N2CCC3(CC2)CC3)=O)CC(F)(F)C1 N1(C(C2(C(=O)OC)CC2C)=O)CCC=C(C(=O)NC2COCCC2(F)F)C1 n1(CC(F)F)nnnc1C1(NCCC2CC2C2CC2)CC(n2cncn2)C1 N(C1CCCn2nccc21)C(C1(CCNC(C(CC)OCC)=O)CCC1)=O c1(OC)noc(C)c1C(=O)NC(CC1CC1)CC(=O)NCC(C)CC1CCC1 N1(C(CCNC(N)=O)=O)CCC2(CCCCC2NC(=O)CCc2csnn2)CC1 CC1CC(=O)NC1C(=O)NCC=C1CCN(C(c2c[nH]c(=N)o2)=O)CC1 N1(C(c2nc(C)cn2C)C(=O)NCCCSC)CC(S(C)(=O)=O)CC1(C)C C(=O)(C(F)C(C)C(F)(F)F)N1C(C)CN(C(=O)C(F)(F)c2cscn2)CC1 C12(C(=O)NC(C(C)C)CNC(=O)CCC3CCCCN3C)CC(C)(C1)OC2C N1(C(c2ccsc2Br)=O)CCc2cccc(-c3ccc(C4CC(N)C4)cc3)c2C1 S(=O)(=O)(c1ccc(N2CCC3(CC2)CC3CO)nc1)NCCCNC C1(CN(C(=O)CC2CCC(O)C2)C)CN(C(c2ccnn2C(C)(C)C)=O)CCO1 c1(CN(CC(c2ccsn2)=O)C)ccc(F)c(F)c1F C1(C(=O)NCCC2N(C(C3C(C)(C)C3)=O)CCOC2)CCCC2C1C2(F)F c1(C(N2C(CNC(Cc3nc(CCC)on3)=O)CC2)=O)nc(O)sc1C c1(C(=O)NC(CC)CNC(=O)CCc2cscn2)cc(O)nc(O)n1 CC1CCN(C(c2ccc(C#N)[nH]2)=O)CCN1C(=O)Cc1cnc2cccnn12 c1(NC(=O)CC2CCCN2Cc2ccc([N+](=O)[O-])o2)cc(Br)cnc1F c1(C(=O)OC)cncc(C(=O)NC2CCC(CNC(=O)CNC=O)C2)c1C N(C)(S(=O)(=O)N(C)C)CC(N1CCC(C)(NC(C=C(C)C(C)(C)C)=O)C1)=O c1(SC)ccc(CCC(=O)NC2(C)CCN(C(=O)C=CC3CCCO3)C2)cc1 N(C(=NCCC(C)C)NCC1(Cc2cccnc2)CC1(C)C)CCS(=O)(=O)NC C(=O)(C1=C(C#N)CCC1)N1CC(CC(C)NC(C2CCCC(=O)O2)=O)C1 C1(CCNCCC2(C(=O)OC)CC2)CCOC(C)C1 c1(C(c2nnnn2C2(C)CC2)NCC(C(CC)C)(C)C)ccnc(P(C)(C)=O)c1 c1(C(=O)NCc2cccc(NC(=O)CC3CC4(CC4)C3)c2)cn2cccnc2n1 CCCCC(CC)CC(=O)N1CC2(CCN(C(=O)CC3SC(=N)NC3=O)C2)C1 Cc1ncc(NC(C2(C)CCCN2C(c2cc3ccoc3s2)=O)=O)c(Cl)n1 c1(C(N(CCCNC(c2ncoc2C2CCCO2)=O)C)=O)cn(C)ccc1=O N1(C(C(CC=C)C)=O)CC(N(C)C(c2cnn(C)c2Br)=O)C2(CC2)C1 C12(CNC(C(CC=C)C)=O)CCC(NC(=O)Cc3cc(F)cc(Cl)c3)(CO1)C2 Cc1nc(C)c(C(N2CC(NC(=O)C3=CCC3)C2)=O)s1 Cc1cc[nH]c(=N)c1C(N1CC(O)(C(C)NC(c2cc(Br)cn2C)=O)C1)=O c1(C(CO)N(C)Cc2n(CCC)ccn2)cccc(Br)c1 C(=O)(CC(C)(C)CNC(C)=O)N1CCC(C)(C(=O)NCc2n(CC)cnc2)C1 C(=O)(CCCC(=O)N(C)C)NCCOCCN(C(C(C(C)C)=C(C)C)=O)C.C(C)(=O)O c1(N(C(COC)C)C)cc(F)cc(F)c1N1CCCC1.C1CO1 CC(C)CC(C)C(=O)NC1C2CC1N(C(=O)CC1CN3CCN1CC3)C2 CC(F)(F)C(C)(C)C(=O)N1CCC(CCNC(C2(c3ccsc3)CC2)=O)CC1 Cc1sc(O)nc1C(=O)NCC1CCCN(Cc2ccc(OCC#N)cc2)C1 N1(C(CCNC(=O)NC)=O)CCC(C)C1C(=O)NCc1ccc(C)s1 C(C1CCN(C(=O)C(C)N2CC(C)C2)CC1)=CC(NOCCC(C)O)=O N1(C(c2ccc(CC#N)cc2)=O)CC2(CCCC2NC(c2cnc[nH]2)=O)C1 C1(C(=O)NC2(CNC(C3N(C)CCOC3)=O)CCCC2)CCc2ncsc2C1 c1(OCCNC(=O)Cn2nnc(=O)[nH]2)ccc(F)cc1Cl C(=O)(CCCCCc1cccs1)N(C1CCN(CCC#N)CC1)C(C(C)C)CO C(=O)(CCC(F)F)NC(C)C(CO)NC(=O)CNC(c1cccnc1)=O C12(C(C(NC(=O)OC(C)(C)C)=O)=O)CCCN(CC1)C2 C1(NC(C(F)=CCC)=O)CN(C(C2CC3C=CC2C3)=O)CC2(CCC2)C1 N1(C(C2(C#C)CCCCC2)=O)CCN(C(c2nccn3ccnc23)=O)CC(C)C1 c1(OC(C)C(=O)NCC2CCCC2NC(C2CC3CC3C2)=O)ccccc1Cl c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CC2)cc(C(C)C)n(C)n1 N1(C(C2(CC#C)CCOC2)=O)CC2C=CC1C(C(=O)N(C)CC1(C)CC1)C2 N1(C(=O)NC(CC)C(=O)O)CCCc2cc(CN(C)C)ccc21 CC1CN(C(c2cc(CCO)on2)=O)CCN1C(c1cc(-c2cccs2)on1)=O c1(CNC(C(C2N(C(CCCOCCC)=O)CCC2)(C)C)=O)ccc(C)cc1O C1(O)(C(N2CCC(N(C(=O)CC3(CS(C)(=O)=O)CC3)C)C2)=O)CCCCC1 c1(C(=O)OC)ccc(S(=O)(=O)NC2=NCCS2)cc1S(=O)(=O)N=c1cc[nH]cc1 CCCC(F)C(=O)N(CCCCCCNC(=O)C#CC1CC1)C C#CCCC(O)C(=O)N1CCN(C)C(CNC(C2CC(O)(C(F)F)C2)=O)C1 CC(C)C1=NOC(C(N2CCC(CCCNC(c3ccc(Cl)o3)=O)CC2)=O)C1 C12(C(=O)NCC(CNC(C3(C)ON=C(C)C3)=O)O)CC3CC1C2C3O N1(C(C2C(F)(F)C23CC3)=O)CCCC2(CCCN2C(=O)CNC(=O)C(F)(F)F)C1 C1(CC(=O)N(C(CC)C(=O)NC2(CO)CC(F)C2)C)C(=O)NN=C1C C=CCC(C)(CC)C(=O)NCCOCCN(C)C(c1cscc1F)=O CC1=C(C)CC(C)(C(=O)NCC2CCN(C(C3(OC(C)C)CCC3)=O)C2)CC1 Cc1cc(=O)n(C)nc1C(=O)NCC(C)(CC(C)C)NC(=O)C(C)NS(C)(=O)=O c1(OC)ccc(C2=CCN(C(=O)C(c3cccc(Br)c3C)F)C2)cc1 Cc1cc(C(N2CC(O)CC2C(N2CC(F)C(F)C2)=O)=O)ncc1N CC(CC(=O)NCC1(O)CCCN(C(c2ccn(C(F)F)n2)=O)C1)P(C)(C)=O N1(C(COc2cccc(C)c2)=O)CC23CCCC2(C1)CN(C(=O)CC1CCC1)C3 c1(C(N2CCC(C3N(C(C(COC)C)=O)CCC3)C2)=O)coc2c(C)cccc12 c1(C(=O)NC(C)(C)CNC(c2ccn(C3CC3)n2)=O)ccc2c(c1)CCCS2 C(=O)(C1CCCc2ncccc21)NCCC1CC(NC(C(C=C)(C)CC)=O)C1 Cc1cnsc1C(=O)NC1(C)CC(C(=O)NCCC2COCCO2)C1 CCCCCC(C)(C)C(=O)NC(CNC(=O)C(O)CC(C)(C)C)C1CCC1 C(=O)(C1CCCc2nccn21)NCCCCC(=O)NCCn1cc(CN(C)C)nn1 N1(C(CCC(C)N(C)C)=O)CCOCC(NC(=O)C(F)=C2CCC2)C1 c1(C(N2C3(CN(c4nc(-c5cccs5)cc(C)n4)C3)CC2)=O)nccc2[nH]ccc12 C#Cc1cc(C(=O)NCC2(CCNC(c3ccnnc3O)=O)CC2)cc(F)c1 c1(CNC(C(N2CCCC2)C)=O)cc(C(=O)N(C2COCCO2)C2CC2)co1 N1(CC(N2CCCCC2Cc2ccnn2C)=O)CC(N(CC)CC)CC1C CC1CC(N(C(=O)C(C)(C)CNC(c2ccnnc2)=O)C)CC(C)C1 c1(C(=O)NC2CC3CN(C(=O)C(F)(F)c4cscn4)CC23)ccnc2[nH]cnc12 c1(NC)nc(C)ccc1C(N1CCC(C)(NC(c2ccc(Cl)cn2)=O)C1)=O n1(CC(C)NC(=O)CCN2CCCC2)cc(CCCC#N)nn1 N1(C(c2c(CNC(=O)CC3CC4(CC4)CO3)cco2)=O)CCN2CCCCC2C1 CCCC(CNC(=O)CCCCNC(=O)CC1(C)CCOCC1)CCO CCC1=C(C(=O)N2CCC(C(=O)NOC(C3CC3)C3CC3)C23CCC3)CCCO1 C(=O)(C1Cc2ccc(F)cc21)N1CCN(C2CCN(C(C(C(=C)C)(C)C)=O)CC2)C1 c1(OC)ccc(NC(C2(C(C)NC(c3cc(Cl)c(C)s3)=O)CC2)=O)cn1 Cn1ccc(CC(=O)N(CCCO)CCCO)c1.C(CC(=O)N1CC(CCCCC)C1)S C(=O)(C(CCCO)c1ccccc1)N(C)CC1(NC(C2CCCS2)=O)CC1 Cc1ccc(OC(C)C(=O)NCCN(CC(C)O)C(c2cc(CO)on2)=O)cc1 c1(C(N2CCC(CC)(NC(C3CCCC3OC)=O)CC2)=O)coc2ccccc12 C1(C(=O)OCC)OCCOC1C(=O)N(C)CCNC(=O)C(C)Cc1ccnn1C c1(N2CCC(CNC(c3c(C)noc3C(F)F)=O)C23CC3)ncnc2scnc12 C(c1cc(Br)cs1)=CC(=O)NCC(C)NC(C1(CO)CCCC1)=O c1(NC(C2N(C(c3ccc(CC)s3)=O)CC(F)C2)=O)cnc(C)c(C#N)c1 O=C1CCCC(c2cn(C3CCC4CC34)nn2)C1.C1(C2N3CC2C3)CCCCCC1 c1(C(=O)NCCC(CNC(C2CCC2C)=O)OC)ccncc1F c1(C(=O)NC2C(NC(C3CC(OC(C)(C)C)C3)=O)C2)[nH]cc2c1CCS2(=O)=O C(=O)(Nn1ccccc1=O)c1cnc(CNC(C(C)C2CCC2)=O)nc1 C1(N(C(C(F)=CC)=O)C)CCN(C(=O)CCOC(C)CC(C)C)CC1 c1(C(N2C(C(=O)NCc3ccc(Br)cc3Cl)CC2)=O)cccc2cncn12 N1(CCNC(CCC)=O)CCCN(C(=O)CCC2(C)CC2(F)F)CC1 N1(C(C(C)C(F)F)=O)CC2CCC(C1)C(NC(=O)CN1CC3CC3C1)C2 N1(C(C2CC(CNC(C3COCCO3)=O)C2)=O)C2CCC1CC(F)C2 c1(C(=O)Nc2cc(CC)c(Cl)nc2)ccc(OC)c2occc12 n1(CC(=O)NC(C(=O)NCC(C)OCCO)C2(C)CC2)ncccc1=O c1(CC)cc(C(=O)NC(C)CN(C(=O)CCc2nnc(S)nc2O)C)c(C)nn1 CCC(C)C(=O)N1CCCC1CN(C(=O)Cc1nccs1)C c1(COCCOCCOCC=C)ccc2c(c1)CCC2 C(C(=O)N1CCCCC1CN(C)C(c1cnsc1C)=O)(C(C)(C)C)NC(C)=O Cc1cc(C)n(C(C)CC(=O)NCC2CCN2Cc2nccs2)n1 c1(CC)ccc(C(N2CCCC2CNS(C)(=O)=O)C(=O)NC2CCOC2)cc1 CC1(C(=O)NCCc2n[nH]cc2C(=O)N(C2CCCCCC2)C2CC2)CCC(=O)N1 c1(C(N2CC(C(N)=O)(CNC(c3c(CCC)nns3)=O)C2)=O)nccc(C)c1N N1(C(c2scc(OC)c2)=O)CCC2CN(C(=O)Cc3cc[nH]n3)C2C1 N1(C(Cc2n(C(C)C)cnn2)=O)CCCC(N(C)C(c2cc(F)n(C)n2)=O)CC1 c1(OC)ccc(Br)cc1COC(=O)NC(=O)NCCCOC1CC1 CC(C)C(O)C(C)(C)C(=O)N1CCC(N(C)C(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C1 c12ccc(cn1)c(=O)[nH]2.N1(CCCN(C)C)CCC(CC2CCCC2)CC1 c1(C(=O)NCC2CN(C(C34CCC(CF)(C3)OC4)=O)C2)nc2ccccc2[nH]1 Cc1ccc(C(C)C)cc1C(=O)NC(C1CN(C(C2(CC3CC3)CC2)=O)CCO1)C N1(C(C(c2scc(C)n2)C)=O)CCCC(NC(c2cc(C(C)C)on2)=O)CCC1 C(=O)(CCC(F)(F)C(F)(F)F)N1C(C)CC(NC(C2(C(F)(F)F)CC=CC2)=O)C1 Cc1ccc(C2CC2C(=O)NCCCCNC(=O)CCc2ccnn2C)cc1Cl C(N=c1[nH]nc(C(C)(C)C)o1)C1CCCN(C(c2cn(CC(C)C)nc2)=O)C1 CN1CCN(Cc2c(NCc3ccc(-c4ncccn4)cc3)cccc2)CC1 Cc1cnc(CN2CCC(O)C2C(=O)Nc2cc(-c3cccs3)nn2C)cc1Br CN1CC(NC(c2conc2CNC(C2CC3(CCC3)CO2)=O)=O)C(F)(F)C1 C1(CNC(C(C)C#N)=O)CN(C)CCN1C(c1cc2ccsc2s1)=O CC1C(NC(=O)Cc2c(F)cccc2F)CCCN1C(c1cccc(N)n1)=O C1(C(=O)NCCCNC(c2cc[nH]c2-c2ccccc2)=O)CCCC(CF)C1 N1(C(=O)CCN2CCCCC2)CCCC(CNCc2ccsc2Br)C1 N=S(=O)(CC)c1ccccc1.N1(C(=O)C(F)Cl)CC(F)(F)CC1c1ccc(F)cc1 c1(OC(C)C(=O)N(C)CCN(C(C2CCCN2C)=O)CCO)ccccc1 N1(C(C2(OC)CCC(C)C2)=O)CCC(C(N2CC3(CCC3O)C2)=O)CC1(C)C C(=O)(CCC(=O)N(C)C(C)C)NC1C(NC(c2cc(C(=O)OC)[nH]c2)=O)C1 c1(CN2C(C)(C)CN(C(=O)CC3CCCNC3=O)CC2)c(Br)cc(F)c(F)c1F C12(C(N3CCC(CC(C)NC(=O)C=CC4CC4)CC3)=O)CCC(CC1)CC2 CCS(=O)(=O)CCNC(C1CCCN(C(C2CCC(=O)O2)=O)C1)=O c1(C(=O)NCC(CC=C)NC(CCCCC#C)=O)cn(C)c(=O)c(C)n1 CC1(C2CCCN2)CCN(NC(C2(O)CCCCC2)=O)C1 c1(C(=O)NC2C(NC(Cc3n(C)cnc3)=O)CCC2)c(Br)ncn1C C1(C(=O)OC)C2CC1N(C(c1ccccc1-n1cccn1)=O)C2 CC1(C)CC(NC(c2ccsc2)=O)CCN(C(=O)CCCC2CCCCC2)C1 C12(CNC(c3nc(OCC)sn3)=O)CCC(CC1)N2C(C1CCCS1)=O C#CCC(C(=O)N(CC(C)(C)CNC(c1ccc(C(=O)SC)cc1)=O)C)C1CC1 C(CCC(C)(c1nnnn1C(C)(C)CC)NC1(C2CCCCO2)CC1)OC CC1CCN(C(C2(C)CCCCC2C)=O)CC1CC(=O)NC(CO)C(N)=O c1(SCCCC)ccc(C(=O)NC(C)Cn2cc(CC3(n4ccnn4)CC3)nn2)o1 N1(C(c2c(CC(=O)OC)occ2)=O)CC2(CCC2CNC(=O)C=CC(=O)N(C)C)C1 CCC(C)C(C)CNC(C1(N(C(=O)C(C)SC)C)CC1)=O C(=O)(C1OCCc2cc(O)ccc21)NCCN(C(CCCCC=C)=O)C c1(CC)nnc2cc(N3CC(NC(C45CCCCC4C5(F)F)=O)C(C)C3)ncn12 Cc1cc(C(N2CC(CNC(c3sc(N(C)C)nc3C)=O)C2)=O)n(C)n1 C1(C(=O)NC(C(C)F)C)CC(NC(c2cc(C3CC3)[nH]n2)=O)C1(C)C c1(C(N2CCCC(F)(CNC(c3cncnc3)=O)C2)=O)nc(O)nc(O)c1F C(CC1C(=O)NCCC(=O)NCC(O)C(=O)N1)=CC.C(=O)(COC)OC c1(C(=O)NC2CCOCC2NC(c2ccns2)=O)cc2ccc(Cl)cc2s1 c1(NC(C(CN(C)C)NC(CCC#CC)=O)=O)c(O)cccc1F CCCC(CC)CC(=O)N1CC(NC(=O)Cc2csc(-c3ccsc3)n2)C1 c1(CO)ccc(C(=O)NC(Cn2cccn2)C(=O)NCC2(CC)CC(F)C2)cn1 C1(NC(C(c2ccnn2C)C)=O)CCN(C(=O)CC(C)F)C1C(C)(C)C C(CCCCCCC)NCC(CC)Cc1ccc(Cl)cc1.O1NC(=O)NCC1 C(=O)(C1=C(Cl)CCOC1)NCCC(C)N(C(C(CC)SC)=O)C C123CCC(CC1)(C2)NC3=O.n1(CC(=O)N)cncn1.C=CCNC(=O)NCC=C [N-]=[N+]=NCCCC(=O)NC1CCCCC1CNC(=O)CC(c1cccc(F)c1)O CC1(C(=O)NCCCNC(c2ccc(OC(F)(F)F)nc2)=O)CC2C=CC1C2 C1(CCNC(CSCCOC)=O)CCN(C(c2cccc(C)c2F)=O)CC1(F)F CCC(CC1CCCCC1)C(=O)N1CCCCC1CN(C(=O)C1=NOCC1)C C(C(C)(C)CN=c1ccnc(NCc2ccnc(OC(F)F)c2)[nH]1)OCC Cn1cc2c(n1)CC(c1nc(CC3CCOC4(CCOCC4)C3)no1)NC2=O c1(CCC(=O)N(CCC)Cc2ccccc2)ccc2cnn(C)c2c1 n1(C(C)C)nc(Cc2cccs2)nc1-c1cnn(C)c1 CC1CN(C(c2cnn(-c3ccc(F)cc3)c2)=O)CC(C)C1NC(=O)C1CC1 CC(O)C(F)(F)C(=O)NCC1CN(C(=O)C(c2cccc(F)c2)O)C1 c1(CC)ccc(C(=O)NCC(C)(C2CC2)NC(=O)CCc2cnc[nH]2)cc1Cl c1(OC)ccc(C(=O)NC(C)CC(C)NC(C2(CF)CC3(CCC3)C2)=O)c(C)n1 c1(C(=O)NC(CN(C(c2ccon2)=O)CC)C)cc(F)cc(N)c1F c1(C(C(=O)NCC2CC2)N(CC)Cc2ccoc2)csc(Br)c1 N1(C(Cn2nc(C)oc2=O)=O)CCC(NC(=O)CC2CS(=O)(=O)C2)C(C)(C)C1 C(=O)(CC(CC)C(C)C)NC1C(C)CN(CC)CC1C.c1(NC=O)ccnc(N)n1 O=C(C(O)C(F)(F)F)NC(C(=O)NCC1CC12CCOCC2)c1ccco1 C12(NC(C3CCC(NC(C)=O)C3)=O)CCCC1N(C(C1CCCC13CCC3)=O)CC2 CC(C(=O)NCC(C(=O)N1CCC(C)(F)C1)C(C)C)S(N)(=O)=O Cn1nc(C(=O)NCC2(CNC(c3ccn(C)n3)=O)CCC2)cc1OCC(F)F CC1CCCC=C1C(=O)NCC(C)C(F)C(=O)NCCCc1ccco1 c1(C(=O)NCCCNC(C(CC)(C)C)=O)cc([N+](=O)[O-])ccc1SCCO N1(C(c2c(SC)cccc2)=O)CCC(C)(CNCc2c(Br)ccnc2Cl)CC1 Cn1nc2c(c1NC(c1sccc1NS(=O)(=O)CCBr)=O)CCC2 C1(NC(C(C)(C)C2CCOCC2)=O)COCCN(C(=O)Cc2csnn2)C1 CC1CN(C(=O)C(C)(C)c2cscn2)CCN1C(=O)CC1CCC(=O)O1 N1(C(C(c2ccccc2)NC(c2c(NC)cccc2)=O)=O)CC2CCCCC2C1 c1(NC(N(C)CC2(C)CC2(F)Cl)=O)ncc(Cl)c(-c2ccccc2)n1 N1(C(C2C(C(=O)OC)C2)=O)CCC(C2CCCN(C(=O)Cc3nocc3C)C2)C1 N1(C(C)C)CCCC1c1nccn1C(C)(C)C.c12ccc(o1)CN(C(C)C)C(=O)N2 C1(NC(CCc2cc(C)[nH]n2)=O)CN(C(C2(CO)CCCO2)=O)CC2(CC2)C1 C(=O)(C(C)CC(C)C(C)=O)NC(CC(CC)C)C(=O)NCc1ccco1 C(=O)(C(C)C(C)C)N.N1(CC)CCOCC1.N12CC(C1)NC(=O)N(C1CC1)CC2=O c1(C(=O)NC(Cn2cncn2)C(=O)NCc2cscn2)ccc(F)c(O)c1 N1(C(C2(CC=C)CC2)=O)C2CCC1CC(NC(C1CC(C#N)(OC)C1)=O)C2 CCCCC(C)C(=O)NCCCCC1CN(C(=O)C=NOC)C1 N1(C(C(N2CC3(C)CCN(C)CC3C2)=O)=O)CCCC(C2CCOCC2)C1 c1(C(=O)NC(C)CCNC(=O)CCn2ccnn2)csc2nnsc12 C1(C)(NC(CCC(=O)OCC)=O)COc2ccccc21 C=C(C)C1OCCC1C(=O)N(C(CC(F)F)C(=O)NCc1ncc[nH]1)C c1(NC)ccc(C(N2CCN(C(C3CC3CF)=O)CC2C)=O)cc1[N+](=O)[O-] CC1=NOC2(C1)CC(C(N1CCCC(CO)(CNC(c3ccsc3)=O)C1)=O)C2 c1(C(=O)NC2CN(C(c3ccc(C)cn3)=O)CC2F)ccc(Br)cc1C(F)(F)F c1(C(=O)NCC2OCCC(NC(Cc3cc(C)[nH]n3)=O)C2)nc2c(s1)CCCC2 C(=O)(C(C)C(O)CC(C)C)NC(CC(=O)NC(COCC)C)CC(C)C N1(C(c2cn(C)nc2C(F)F)=O)CC2(CC(NC(=O)C#CC3CCCO3)CO2)C1 c1(OC)cc(C(N2CCOC(C)(CNC(c3ccc(SC)s3)=O)C2)=O)ccc1C C(c1ccc(Cl)cc1)=CC(N1CC(NC(C(C)C2CC2)=O)C(C)C1)=O C1(NC(COC2(C#C)COC2)=O)CC12CCOCC2 c1(C(=O)NC2CN(C(COCC)=O)C(C)C2)cc(NS(C)=O)ccc1F c1(SC)cc(C(=O)NC2CCC2CNC(=O)CCc2nc[nH]n2)oc1C C(CC(C)C)(CC(C)C)NC(C(C)NC(C1C(OC)CCC1)=O)=O C(=O)(C(C(C)C)OC(F)F)NC(C(c1ccccc1)OC)C c1(CCC(=O)NC2C(NC(C(C)c3ccsn3)=O)CC2)ccc(Cl)cc1 Cc1nc2c([nH]1)CC(C(=O)NCCCCCNC(c1ccc(Cl)c(C)c1)=O)CC2 c1(NC(C(CC2(C)CCOC2)N(C(C#C)C2CCC2)C)=O)ccc(F)cc1C S(=O)(=O)(c1cccc(=NCCCF)[nH]1)NC1c2ccc(C)cc2CCC1 Cc1cc(C(=O)NCC(C)NC(=O)Cc2ccsc2)cc(Cl)n1 c1(C(N(C)CC2(CNC(C3(C=C)CC3)=O)CC2)=O)cnc(O)c(OC)c1 c1(C(C)O)ccc(C(=O)NCC2CCN(C(=O)C(C)(C)N3CCCC3)C2)c(N)c1 c1(C(=O)NCC(N(C(CNC(CC)=O)=O)C)C2CC2)cnn2c1S(=O)(=O)NCC2 C1(CN(C(=O)CC2C3COCC23)C)CN(C(=O)CCN2CCCC2)CCO1 C1(C(N2CCC3CN(C(=O)CC(F)(F)F)C3C2)=O)CCOCC12CCC2 c1(CNC(=O)CC(N)c2ccccc2)ccc(N2CCCC2)cc1 N1(C(C=CCC)=O)CCC(F)(CNC(c2ccc(C3CNC(=O)C3)cc2)=O)CC1 c1(CN2C(CC(=O)Nc3cccc4c3OCO4)CC(F)C2)cc(F)c(Cl)c(F)c1 CC(C)(C(=O)N1CCCOC(CNC(C2(C)CC=CCC2)=O)C1)C(F)F C(C(CC(C)C)C(=O)N(C)C)NC(Cc1c(F)ccc(C)c1)=O N1(C(C=C(CCC)CCC)=O)CCC2CC2(NC(=O)CCCC(N)=O)CC1 c1(OC)ccc(C(=O)NCC(C)(C)NC(=O)CCC(=O)NC2CCCC2)c(F)c1 C1(OC)CN(C(=O)CCOc2cc(C)ccc2C)C2(CCCC2)C1 C(=O)(C(Cc1nccs1)NC(C)=O)NC(CC)COCC(F)(F)F N1(C(c2c(C)nc(COC)s2)=O)CCCC(NC(=O)CCSC(F)(F)F)C(F)C1 N1(C(CC)=O)CC2CN(Cc3c(C)nn(C)c3C)CC12 C1(NC(C(CC)O)=O)CCC(C)N(C(=O)C(F)Cc2ccccc2)C1 c1(NC(C(n2cc(COCCO)nn2)C)=O)cccnc1O C1(C(=O)NCC(C(C)C)NC(=O)C(C)NC=O)CCCOCC1 C(=O)(CC(F)(F)F)NCC(=O)NC1(CNC(CCCNC(C)=O)=O)CCOC1 c1(Cc2nc(-c3cc(CC)c(Cl)cc3)on2)cn2cccc(C)c2n1 C#CC1(C(=O)NC2(CC(=O)OC)CC2)CCN(C(C2CC(CC)C2)=O)CC1 C(=O)(C(F)(CNC(=O)CCCC(F)(F)F)C(C)C)NCCCC=CC c1(C(=O)NCC(CNC(=O)CN(c2ccn(C(C)C)n2)C)OC)ccoc1C C1(C(N(C)CC#N)=O)Cc2c([nH]c3ccccc23)CN1Cc1cc(Br)ccc1Cl c1(OC)cc(C)c(C(=O)NC2CCN(C(c3ccc(C)c(Cl)c3)=O)C2)cn1 c1(C(N2C3CC(C(NCP(C)(C)=O)=O)(C3)C2)=O)cc(F)cc(F)c1 N1(C(COCCC#C)=O)CC2(CCC(NC(C3CC3(C)COC)=O)CC2)C1 c1(CC)c(C(=O)NCC(C2CCC2)NC(=O)C=CC2CCCN2C)cnn1C C1(CNC(C2N(C)CCC2)=O)CC2(CO1)CN(C(=O)Cc1sc(O)nc1O)C2 c1(NC(CC(=O)NCC)=O)ccccc1C1CC1(F)F.C12(CC)CN(C1)C2=O C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)Nc2cc(C)c(O)cc2C)CNC(=O)C1 C1(CNC(=O)CCc2ccccc2F)C2CN(C(=O)Cc3cccc(Cl)c3)CC12 c1(C(N(CCN(C(CN2CC(C)C2)=O)C)C)=O)csc2c1CCCC2 CC(CF)C(=O)N1CCCC1C(C)(C)NC(=O)CC1CC1 CCCCCCC(C)C(=O)NCC1CCN(C(=O)C(CC(C)C)N(C)C)CC1 c1(C(N2CC(CC(=O)NC3C(CC(C)(C)C)C3)C2)=O)cccc2c1OCCCO2 C(C(O)C(=O)N1CC(CC(C)NC(c2cnc(O)o2)=O)C1)OC Cc1cnnc(N2CCC(C)(C)C2CN)c1C C(C(C)(C)CC(=O)N(CCC(=O)NOCc1nncn1C(C)C)C)OC N1(C(C23CC=CC(C2)OC3)=O)CCC2(CC1)CC2c1cn(CC2COC2)nn1 C(C)(N=c1[nH]c2c(c(=NC(C)c3nc(C)cs3)[nH]1)COC2)c1nc(CC)[nH]n1 C1(C(=O)NC2CC(NC(c3csc(-c4cnn[nH]4)n3)=O)C2)(OCC)CCCC1 c1(C(N2CCOCC(C(N3CC(SC(F)F)C3)=O)C2)=O)cc(F)cc(F)c1 N1(C(C(C(C)O)C)=O)CCC(C2CN(C(c3ccccc3P(C)(C)=O)=O)C2)CC1 C1(C(C)NC(CCOC(C)=O)=O)CCN(C(C2CC(C)=NO2)=O)CC1 N1(C(c2ncc(C)c(C)c2)=O)CC2CCCCC2(NC(C23CCCC2C3)=O)C1 N1(C(C(CCC)OC)=O)CC2(CNC(=O)C(C#N)C(C)(C)C)CCC1CC2 c1(OCOC)ccc(-c2ccc(C(=O)OCC3CC(C)C3)nc2)cc1OC C1(C(N(CCNC(C2CCN(C(CCC)=O)C2)=O)CC)=O)CC(C)(C)CN1C N1(Cc2nc(C)oc2)CCNC(c2ccccc2C)C1 C1(C(N2CC(F)(CC)C2)=O)CN(C(c2n[nH]cc2Cl)=O)CC1F CCC(CC)C(C(=O)NCC(COC)NC(c1cccc(C(C)C)c1)=O)OC CC(C1CCCc2ccccc21)n1cc(CCc2ccccc2)nn1 n1(CC)cc(C(=O)NC(C2CCOC2)CNC(C2CC2F)=O)nn1 C1(C(=O)NCC(C)CN(C)C)CCCN(C(c2ccnn2C(F)F)=O)C1 C=C=CC(C)C(=O)NCC(C)(C)CN(C)C(c1ccncc1Br)=O Nc1ccc(C(=O)NC(CNC(=O)C=Cc2cccnc2)C2CCC2)c(O)c1 Cc1ccc(C(=O)NC(C(=O)NC2CCC(F)(F)C2)C2CCCC2)nn1 C(CC(C(=O)N(C)CC1C(C)C1)NC(C1C2CCC(F)C12)=O)Nc1cccnn1 C1(CN(C(C=C=CC=CC)=O)CC)CCCCN1C(=O)COC1CCCC(C)C1 c1(C(=O)NC2COCCN(C(C3(C)CC(=C)C3)=O)C2)cccc2c1NCC(C)C2 C#CC1(C)CCCN(C(C23CCCC2CN(C(C2CSCCS2)=O)C3)=O)C1 C1(NC(C2C(NC(Cn3c(C)ncc3)=O)COCC2)=O)CC2CCC(C1)O2 c1(C(CC)OC)ccc(C(F)(F)F)cc1OC.c1(C2CCC2)noc(C(C)C)n1 CC(C)(C)CC(C)(C)C(=O)NCC1(O)CCN(C(c2cnn(C(F)F)c2)=O)C1 C(=O)(C(C)P(C)(C)=O)N1CCCC(N2CCN(C(c3ccc(C)o3)=O)CC2)C1 N1(Cc2cc(C)no2)CCC2(CC1)OCCC2NC(c1cnnn1C)=O O=S(=O)(c1c[nH]ccc1=NCC1SCCS1)N1CCC2(CC1)OCC1CC21 N1(C(CCCOC)=O)CCC2(CC1)CC(NC(C1CCc3n[nH]cc3C1C)=O)C2 Cc1cccc2c(CNCc3ccc(C=CC(F)(F)F)cc3)n[nH]c12 c1(C2C(C(C)NCc3cnn(CCF)c3)C2)c(Cl)cccc1Cl Cc1nc2cc(C(=O)NC3CC(CNC(=O)C(C)CC(F)(F)F)C3)cnc2s1 C1(CC(=O)NC2COCCC2NC(=O)C2=CSCS2)CN2CCN1CC2 N1(C(CCCOCC)=O)CCC(CO)(NC(=O)CCn2cncn2)CC1.C1(C)CC1 C(C1=NOC2CN(C(c3ccnc(O)c3)=O)CC12)NC(=O)CCF c1(C(N2CC(C(C)NC(=O)C(C)(C)C)OCC2)=O)cc(P(C)(C)=O)ccn1 N=c1[nH]c2cccc(C(N3CCNC3c3ccccc3)=O)c2s1 CC1(C)CCC(N=c2[nH]c(=NC3COc4cccc(Cl)c4C3)[nH]c3ccsc23)C1 c1(C(N2CC(O)(C(C)NC(=O)CCN3CCCCC3=O)C2)=O)c(N)cccc1F C(=O)(CCCCCN=[N+]=[N-])NC(CC#C)C(=O)NCCc1cn[nH]c1 C1(C(N(C(C#C)C2CCC2)C)=O)CCN(C(c2scc(C)c2C)=O)C(C)(C)C1 c1(N(C)C(=O)Nc2ccc(Cl)cc2Cl)cccc(SC(C)(C)C)c1F C1(SC(C)C(=O)NC(CNC(C2CC2c2ccccn2)=O)C2CC2)CCCC(C)C1 CCCC(C)(O)C(=O)NCC1(OC)CN(C(C2(C)CCCC2C)=O)C1 C1(N(CC(=O)NCCCOC)CCCNC(c2ccccc2)=O)CCCOC1.OCC C1(NC(C(CC#C)C2CC2)=O)CN(C(=O)C(C(C)C)C2CCC2)CCC1C n1(CC(=O)N(C)CCNC(=O)CC2CCC(=O)N2)cnc(C#N)n1 c1(C(N2CCC(NC(=O)Cn3nccn3)CC2C2CC2)=O)cc(F)c(F)c(O)c1F c12ccc(cc1)OC2.C1(OCCC(=O)NCCCCl)CCCCC1 c1(C(N(CCN(C(C2CC2(C)CC)=O)CC)CC)=O)csc(-c2csc(C)n2)c1 C1(O)(CC#C)CC(C(=O)NC(C)(CNC(c2cnn(CCl)c2)=O)CO)C1.C(C)(C)(C)O C1(OC)CCCCC1C(=O)NCCCC(C)(C)NC(c1nc(C2CC2)cs1)=O Cc1ccc(C(N2CC(OCCNC(C34CC(C(F)F)(CO3)C4)=O)C2)=O)cc1F Cc1ccc(-n2cc(CN)nn2)c(Br)c1.C1(C(=O)N)CC(=C2CCC2)C1.C1CS1 CCC(CCC(=O)N1CCN(C(c2cc(N)ccc2O)=O)C(C)C1)OC c1(OC)cc(CO)ccc1C(=O)NCC(C(C)C(C)C)NC(=O)C=C(C)C(F)F C1(C(=O)NCC2(C(N)=O)CN(C(c3cnn(CC)n3)=O)C2)CC(C(N)=O)CCO1 CC(C)C(C)C(=O)N(CCCNC(=O)CC(C)n1ccnc1)Cc1ccccc1 Cc1cc(C)c(OC(F)F)cc1Br.C1CSCCO1 C1(N2CC3C(CC)(C3)C2)CC2CCC(C1)C2 c1(C(=O)NC2CC(NC(C=CC=CCC)=O)C2)cc(N)c(Cl)cc1F CN(CCc1ccc(F)cc1)N1CCN(C(=O)Nc2ccccn2)CC1 S(=O)(=O)(c1ccccc1)N1C(C)(C(=O)NC2C(C(=O)OC)C2)CCC1 N1(C(c2cnn(C(C)C)c2Cl)=O)CC(NC(C2(C)CCCOC2)=O)CC(F)C1 C1(CC(=O)NCc2cn(CC)nn2)CC2(CC2)CN1C(c1ccc(C#N)cc1)=O c1(C(=O)NC2(c3cccc(C(=O)OC)c3)COC2)nc(C(F)(F)F)oc1C c1(CC(=O)NCCOCCCNC(c2cc[nH]n2)=O)ccccn1 C(=O)(CC(C)CC(C)C)N(C1CC(NC(c2ccc(NC)c(F)c2)=O)C1)C c1(NC(=O)OC)c(C(N2CCC(NC(=O)CN)C(CO)C2)=O)sc2ccccc12 Cc1cnc(SCC(N2CCC(NCC(=O)N)C2)=O)c(C)c1.C1(C(N)=O)CCC1 c1(-c2nc(N3CCN(C(C)=O)CC3)sc2)cc(F)c(O)cc1F C1(NC(c2c(SC)n(C)nc2)=O)CCN(C(=O)C(C)(C)CF)CC1CO N1(C=O)CC23CCCCC2(COC3)C1.C1CC2CCCC(C1)C2 N1(C(c2cc(O)nc(O)n2)=O)Cc2cccc(Cl)c2C1.C12CC1C(=O)N(C)C2=O C1(NC2CC(O)C2)CCN(C)C1.CC(CCOC(C)(C)C)NC(C)(C)C C1(N(C)C(C2CCCN2C(N)=O)=O)CCCCN(C(c2ccsc2)=O)C1 CC1CC(C(N2CC(C(N)=O)(CNC(=O)CC3CCN(C)CC3)C2)=O)CC(C)C1 C1(C)(NC(=O)OC)CCCCC1C(=O)NCc1ccc(Cl)cn1.C1C(=O)N1 C(N=c1[nH]c(=NCC(=O)N2CCCO2)[nH]c2c1CC(C)(C)C2)C1(CS(C)(=O)=O)CC1 n1(CC(=O)NC2CC(OCC(=O)NCCCCNC)C2)nnc(C)n1 N1(CCCNC(c2c(-c3cn(C)nc3)cco2)=O)CCN(c2ccccc2)CC1 c1(C(N2CC(C#N)C(NC(C3CCCS3)=O)C2)=O)cc(=O)c2ccccc2o1 c1(C(=O)NC2CC(C)N(C(c3cccc4c3OCO4)=O)C2)cc2n(n1)CC(F)C2 N(C(=NCCC1(O)CCC1)N1CCC(C(F)F)C1)C(COC)C C1(Nc2ccnc(C)n2)CN(C(=O)C2=CCCCC2)CCC1F c1(C(COC)NC(=O)Cc2nc(C(=O)OC)cs2)cccc(C)c1 c1(C(N2C(CNC(c3ccn(CC(F)(F)F)n3)=O)C=CC2)=O)cncc(Cl)c1 c1(C(N(CC(C)NC(C2CC(C(=O)OC)C2)=O)CC)=O)cc(C(C)C)on1 C(C(C)(C)N=c1[nH]nc(C(C)(C)C)o1)NC(C(CC(C)C)C(N)=O)=O C(=O)(C1CCCc2nc[nH]c21)NC12C(CN(C(C3(C#N)CC3)=O)C1)C2 C1(C(=O)NC(CNC(C(C)(C)CF)=O)C2CCC2)CC2C=CC1CCC2 C1(c2ccc(CC(C)C)s2)NC(=O)N(CC2CC2)C2=C1C(=O)NCC(C)C2 c1(OC)coc(C(=O)NCCC(C)N(C(=O)C(C)(C)c2ccncc2)C)cc1=O c1(CNC(C(n2cc(NS(C)(=O)=O)nn2)C)=O)cccc(C#N)c1 N1(C(C2(CC)CCCN2C(=O)COCCCOC)=O)CCNC(=O)CC1C N1(C(C2(CC(C)C)CC2)=O)CC(C)CN(C(c2c[nH]nc2Br)=O)C(C)C1 C1(SC)CCC(C(N2CCC(OCC(C)C)C2)C(=O)NCC(C)C)C1 C1(CNC(Cc2c(C)cccn2)=O)CCCCCN1C(=O)C(C)OCC(F)(F)F Cc1ccc(C(=O)NC(C)CCNC(C2(C)CC2(Cl)Cl)=O)c(C)n1 c1(C(=O)NC(C)CCNC(c2cscc2Cl)=O)cnn(C)c1-n1cccc1 c1(C(=O)NC(CC)CNC(c2c(C(C)C)n[nH]c2C)=O)nc(C2CC2)ncc1Cl N1(C(c2c(F)cccc2Cl)=O)CCN(C(C2CCO2)=O)CC2(CC2)C1 C(C)(CCCCNC(C1(n2cccn2)CCC1)=O)NC(C1CCN(C(C)C)C1)=O c1(C(=O)NCC(CN(C(COCCC)=O)C)(C)C)nnc(S)n1C N1(CC(=O)N(CC(=O)NCC2CC2)C)CCNC(=O)C1.C1(C(=O)N)(CCF)CCC1 N1(C(=O)Nc2cc(C)c(N3CCSCC3)cc2)CC(CO)OC2(CCCOC2)C1 C1(CNC(c2ccn(CC)n2)=O)CCCCN1C(=O)C(C(C)C)N1CCCCC1 C1(NC(C(COC)C)=O)CCC2CN(C(c3nncs3)=O)CCC2C1 S(=O)(=O)(c1cccnc1)N1C(C(=O)Nc2ccc(C)cn2)CCCC1 C1(CNC(C(C)OCC)=O)CCN(C(C2CCC=CO2)=O)C1(C)C C1CCCN(C(=O)CCc2ncc[nH]2)C1.C(=O)(C(C)(C)c1cn(CC)nn1)OC C(=O)(C(C)(CC)C(=O)NC(C)CNC(c1ccc(C(F)(F)F)c(N)c1)=O)OCC C1(F)(CNC(c2cnc(CC)s2)=O)CCC(NC(c2ccccc2C2CC2)=O)C1 N1(C(CC(C)OC)=O)CCC2(CC1)CN(C(c1cnc(S)nc1)=O)CC2CO N1(C(CN(C2CC2)CC)=O)CCOC(CSc2cc(CC(C)C)c[nH]2)C1 NC(=O)CCC(=O)NCC1CC(O)CN1C(C1C(F)(F)C12CC2)=O N1(C(C2(OC)CCSC2)=O)CCC(C2CCN(C(C3CC(C)(C)C3)=O)CC2)CC1 C1(C(=O)O)N(C(=O)Cn2cc(CC3CCOC3)nn2)CC12CCCC2 Cc1cccc(C(O)C(=O)NC2CN(C(c3ccc(CO)o3)=O)CC2O)c1 c1(C(COC(C2(c3ccccc3)CCC(=O)NC2)=O)=O)c[nH]c2ncccc12 N1(c2c([N+](=O)[O-])cn(CC)n2)CCC2(CC1)OCCC2NC(=O)CN(C)C Cc1cc([N+](=O)[O-])cnc1C(=O)NCc1cnc(C)n1C c1(-c2cn(-c3cc(C(=O)OC)sc3)nn2)cnccc1NC(c1ccnn1C)=O C(=O)(CC(C)(C)C(C)(F)F)N1CC(C)C(NC(CCCCOCC)=O)C(C)C1 N1(C(CC(C)C(F)F)=O)CC2CCC(CNC(=O)CCC3CCCO3)C2C1 N1(c2n(CC(COC)O)nnn2)CCN(c2ccc(OC(F)F)cc2)CC1 c1(C(=O)NC(CNC(C(CN(CC)CC)F)=O)(C)C)cccc(S(=O)(=O)NC)c1 c1(C(N2C(C(N3C(C(C)C)COCC3)=O)CC3CC32)=O)c(C#N)cnn1C Cc1cn(C)cc1C(N1CCC(C(C)NC(=O)CCCn2ccnc2)CC1)=O C12(NC(=O)NCC3CC(OC)(OC)C3)CCCC1(CO)C2 c1(C(N(CC=C)Cc2cn(CCCC(=O)O)nn2)=O)cc(S(C)(=O)=O)cnc1O C1(NC(COCCCC(C)C)=O)CC2CC1N(C(=O)CSc1n[nH]c(O)n1)C2 C1(C(=O)NCC(COC)NC(=O)C(Cl)=CCl)CCC(=O)N1 N1(C(c2n(C=C)ncc2)=O)CCC2CCC(C1)N2C(c1scnc1COC)=O N1(CC(=O)N(c2ccc(CN(C)C)cc2)CC)CCC(C)(O)CC1.CCSCC N1(C(C(C)Cc2ccccc2)=O)CC2(NC(=O)CN3CSCC3=O)CC1C2 C1(C#N)(C(=O)NCC2CC(C)(C)C2)CC2CCC1C2 C1(NC(CSCC)=O)CCN(C(c2ccc(N3CCC(C)C3)cc2)=O)C12CC2 C1(NC(c2c(CC)cco2)=O)C2CC3C1C3C2C(N1CCC(F)CC1)=O CCC(CC(=O)N(C1CCN(c2nnc(C(N)=O)s2)C1)CC)C1CCC1 C1(NC(C2CCCO2)=O)COC2(C1)CN(C(C1(c3ccccc3)CC3(CC3)C1)=O)C2 c1(C(=O)NC(C2CCCN2C(C2CCCCC2C)=O)C)ncc([N+](=O)[O-])n1C C(CC(C)(C)CC(=O)N(CC(=O)N(C1CCC1)CCO)C)OC.C(CCO)SC c1(NCCC2N(C)CCC2)nc2ccc(Cl)cc2c(=NCCC2(C)CCCO2)[nH]1 C(=O)(C(C(C)c1ccc(Cl)cc1)N(C)CC1CCCCC1O)NC C(CC)(CCCC(=O)N1CCC(N2CCCC2)C1)NC(CC(=O)NCC#C)=O C1(CCC)CN(C(=O)Cc2scnc2C)CCN1C(=O)COCCOC C(CCC(c1nnnn1CC(F)F)NCCNC(=O)CC(C)C)OC C1(C(N(C)CC2(O)CCOC2)=O)CCN(C(=O)COC2CCCCC2)C12CC2 C1(CC)CC(C)CN1C(C1(CO)CCN(C(=O)C=CCOC)C1)=O C(=O)(C(C)CC(=O)N1CSCC1C(=O)NC1CC(F)(F)C1(C)C)OC c1(CCCNC(CN(C(=O)C(C)C2CCOC2)CCOC)=O)nncs1 C1(CC)CN(C(=O)C(C2CC2)OC)CC1CNC(=O)C(C1CC(F)(F)C1)O C(=O)(CN=c1[nH]c(N2CCC(n3cccn3)C2)nc2c1CCCC2)NCC C(CC(C)(C)CC(=O)N1CCC(NC(c2cc(CC(C)C)[nH]n2)=O)C1)OC C12(CNC(C(C)CN(C)C)=O)CC(C(N)=O)(C1)C1(CN(C(=O)CC(C)(C)C)C1)O2 C(=O)(CCCC(=O)N(C)C)N(CCC(=O)N(CC(O)C1CC1)C)CCC c1(NC(C)C(N2CC(Cc3ccccn3)C(O)C2)=O)ccn2ncc(Br)c2n1 C1(CCNC(=O)C=Cc2ccncc2)CN(C(C2CC3(CC3)C2)=O)CCS1(=O)=O c1(C(=O)NC2C(NC(Cn3ncc(C#N)c3)=O)C2)cc2ccnc(Cl)c2[nH]1 c1(C(=O)NCC2N(C(c3ccc(C)cc3C)=O)CCC2)c(C)c(C)cc(C)c1C Cc1nc(O)[nH]c1C(N1CCN(C(=O)C(C)Cc2ccccc2)CC1)=O Cc1cc(C(N2CC(c3noc(C(=O)O)n3)C2)=O)c(C)[nH]1 C(CC(O)C(=O)NCc1cc(C(N)=O)co1)NC(C(C)(O)C1CCC1)=O CC1Oc2ccc(CN3CCCC3CC(c3ccccc3)O)cc2NC1=O C1(C(=O)NCC2(O)CN(C(C(C)OCC(C)C)=O)C2)OCCN(C)C1=O N1(C(C(C#N)=CC(C)C)=O)CC(N(C(=O)CP(C)(C)=O)C)C2(CC2)C1 C1(C(=O)NC(c2cn(Cc3nc(C(N)=O)cs3)nn2)C)CCC2(CC2)C1 C1(NC(=O)NCCCOC)CCS(=O)(=O)C12CN(C(=O)CC1(C)CCCC1)C2 C(=O)(C(C)(C)CS(N)(=O)=O)NC(C1CCN(C(c2n[nH]c(C)c2F)=O)C1)C C(=O)(CCC(=O)NCC(CC(C)C)NC(c1cnc(COC)nc1)=O)NCCC Cc1[nH]nc2ncc(C(=O)NC3CN(C(c4ccccn4)=O)CC(C)(C)C3)cc12 c1(C(=O)NC2CC(NC(CC(C)CN(C)C)=O)CC2O)cc2c(Cl)cccc2[nH]1 N1(C(COC)=O)CCc2c(CNC(C3CCCN(S(C)(=O)=O)C3)=O)cccc2C1 c1(CC(=O)NCC(C)=CC(N2CC(C)(C)C2)=O)ccc(C)nc1 CON1CCC(CC(=O)NC2CCCC2NC(c2cc(Cl)ns2)=O)CC1 C12(C(N3CC(CNC(C(C)(C)c4ccccc4)=O)C3)=O)CCCN(CC1)C2 CCC(CCC(=O)N1CCCC(NC(c2oc(CC)cc2C)=O)C1)OC C(=O)(C1c2ccccc2C2CC1C2)NCCC(N=c1nc(C)[nH]n1CC(=O)NC)=O C1(C(=O)NC(C)(C)CC(F)(F)F)CCN(C(=O)C(C(C)(C)C)NC(N)=O)O1 n1(-c2cn(CC)nc2)nc(CCC2CCCO2)nc1-c1cnc(-c2ccco2)s1 N1(C(C2CCCC(C)C2)=O)CCCC(C)(C)C1CNC(=O)C(C1CCCCC1)O N1(C(c2ccc(OC)nc2)=O)CCCN(C(=O)CCCCC2CCCCC2)CC1 c1(NC(=O)CC2CCCC2NC(C23CCCC2CCC3)=O)cnc2c(c1)CCC2 c1(C(=O)NC2CCCC(NC(C3N(C)CCCC3)=O)C2)coc2c1COC2 C1(CNC(CN(CCOC)C)=O)CCN(C(=O)Cc2ccc(Cl)cn2)C(C)C1 CCCC(CC)C(=O)NC1CCN(C(=O)C(F)C2CCOC2)CC1F C(=O)(CC(C(F)(F)F)N1CCOCC1)NCCNC(c1cnc2ccccn12)=O c1(CC)nccn1CC(=O)N(CC(C)NC(C1CC1=C(C)C)=O)C CCS(=O)(=O)CC(C)N(C(=O)Cc1sccc1OC)C c1(C(=O)NC(C2CN(C(=O)C=Cc3cscn3)C2)C)cc(Cl)cnc1O C(=O)(CC1COc2ccccc21)NCCCCN(C(=O)C1=NOC2(CCC2)C1)C C1(C)(C(=O)NCC2CC3N(C(COC(C)=O)=O)C(CC3)C2)CCc2ccccc21 c1(C(=O)NCC(C2CC2)NC(=O)Cc2ccncc2)cc[nH]c2nccc1-2 N1(C(CC2CC(OC)C2)=O)CCCC1CNC(=O)Cc1csnc1C C1(C(=O)NC2CC(NC(C(CC)NC(N)=O)=O)C2)CCCCN1S(N)(=O)=O CCC(C)(C(=O)N(CCNC(=O)C(C)OCC1CCCC1)CCOC)OC C(=O)(CCCCC(F)F)N(CCOCCC(=O)NCCCCC#C)C.C1(=O)CN1 CCC(O)C(C)C(=O)NC1CC(CNC(=O)COCc2cccc(C)c2)C1 c1(C(=O)NCCOC2(C)CN(C(COC)=O)C2)ccc(C#N)c(OC)c1 c1(C(N(CCC)CCNC(=O)CC2CCCC2(F)F)=O)ccc2nc(O)[nH]c2n1 c1(C(c2nnnn2CC2CCOCC2)NCC2(C)CCCO2)ccc(F)cc1Br C1(CC=C)(C(=O)NCC2CCNC(=O)C2)CCN(C(=O)C(n2cc(C)cn2)C)C1 C(=O)(C1=CCCSC1)N(C1CCCC1CNC(c1cc(O)nn1C)=O)C C1(CNC(c2c(C)[nH]nc2C(F)(F)F)=O)CN(C)CCN1C(=O)COCCO N1(C(C2CC(C(=O)OC)C2)=O)CCCc2cc(Br)ccc2C1 N1(C(C2CC(=O)OC2)=O)CCCC(C2CC2NC(C2(CCO)CC2)=O)C1 CCC(COC)(CC)C(=O)NC(C)CC(=O)NCCC(O)CO c1(C(N2CC(O)(CNC(=O)CCC=CBr)C2)=O)cnc2ncccc2c1 C(=O)(CC(C)CC(=O)NCC1CC(F)(CNC(c2ocnc2CC2CC2)=O)C1)OC C1(NC(C(C2CCCCC2)C)=O)CCC(C)(NC(C2CCC3CC23)=O)CC1 C(=O)(C(C)(O)CCN(C)C)N1CCC(C)(NC(c2c(C)nc(C)o2)=O)C1 c1(OC)cc(F)c(C(=O)NCCCC(C)NC(c2ccc(O)nc2)=O)cc1OC c1(C(=O)NC(CCNC(C(CC)OC)=O)Cc2ccccc2)ccc(OC)nn1 Cc1ccc2[nH]nc(C(N3CCOC(CN(C(=O)CC(C)C(F)F)C)C3)=O)c2c1 C(CN=c1[nH]c(=NCC#Cc2cnn(C)c2)c2ccccc2[nH]1)C1(OC)CCC1 n1(COC)ncc(C(=O)NC2(CCCCNC(C3CCCC(F)C3)=O)CC2)c1C C1(C(N2CCC(CNC(C3CC(C(C)C)C3)=O)C2)=O)(CC)CCCCC1 CC1(CNC(=O)CCc2cnc[nH]2)CCN(C(=O)CNC2CCCC2(F)F)C1 C(=O)(CC(F)(F)C(C)(F)F)NC(C)CCCNC(=O)C(c1ccccc1)F c1(C(N2C(C)(C(=O)Nc3c(C(=O)OC)csc3)CC2)=O)c(O)c(Cl)cc(Cl)c1Cl C(CN=c1cc[nH]c(=NCCc2cccnc2C)[nH]1)(C(C)(C)C)SC CN1CC=CCC1CC(=O)NC1CCC(CC(=O)NCc2cncc(Cl)c2)C1 Cc1nc(C(F)(F)F)oc1C(=O)NC1(C)CCN(C(C2CSCCS2)=O)C1 N1(C(c2cc(Br)no2)C(=O)NC2(C)CC2)CC2CCC(CC2)C1 C=CCCCCCN(C(c1sc(Br)cc1Cl)C(=O)NC1CCCC1)C Cc1nc2sccn2c1C(N1CCCC1CNC(=O)C(C)c1ccco1)=O n1(C(C)C)cnc(C(=O)NCCCCCN(C)C(c2cnn(C)c2)=O)c1 C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)CN2C(=O)CCC2=O)CC12CCC2 CC(C(=O)NC1CC12CCN(C(C1CCCN1N=O)=O)C2)S(N)(=O)=O c1(OCCOCC2CC2)ccccc1C=CC(=O)NN1CCNC(=O)C1.N1(CC)CCC1 c1(C(=O)NC(CCC)CNC(=O)C(F)(F)CC)cncc2nc(C)[nH]c12 c1(C(=O)NC2C(NC(=O)C=CCc3cccnc3)C2)cccnc1-c1ccccc1 c1(C(N2C(CNC(c3cncc(N(C)C)c3)=O)CC2)=O)scc2c1OCCO2 C1(N(C(c2ncn(CC)c2)=O)C)CCCC(NC(C2(CO)CCCCC2)=O)C1 c1(C(N(CC)CC2CCN(C(c3n[nH]cc3Br)=O)CC2)=O)ccc(O)c(O)c1 N1(CC(=O)NCC2(CNC(c3cocn3)=O)CC2)CCSC2CCCCC12 Cc1c(CNC(=O)NCC2C(Sc3ccccc3)C2)noc1-c1ccc(Cl)cc1 Cc1nc2ncccc2cc1CC(=O)N(CCCNC(=O)CCS(C)(=O)=O)C1CC1 C1(CNC(=O)CC2CCCCO2)CCCCN1C(C1CCCCCC1)=O C1(C(=O)NCC2CCC2C(=O)NCCCO)CNC(=O)O1 c1(C(=O)NC2CC(NC(C(C(C)C)(C)C)=O)C2)cc(Br)c2[nH]cnc2c1 N1(C(=O)CCCCCO)CCCC2(CCCN2C(=O)C2CCCc3ccnn32)C1 C(=O)(CCCCCC#N)NC1C(C)(C)C(CC(=O)NCC2=NOC3CCCC23)C1 Cc1c(CC(N2CCN(C(C3CC=CCC3C(F)(F)F)=O)CC2)=O)ncn1C C1(C(=O)NC(C2(O)CCCC2)C)COC2(C1)CN(C(=O)CC1(O)CCCCC1)C2 N1(C(c2c(C#C)c[nH]n2)=O)CC(O)CC1(C)C(N1CC2(CCCO2)C1)=O c1(C(=O)NC2CN(C(c3ncc(C)cc3Br)=O)CC2F)cccc2ccncc12 c1(NC(C2(C)CN(Cc3n(CC)ccn3)C2)=O)nc(O)nc(O)n1 N1(CCOC)C(=O)CC(C(=O)NCC(C2CCOCC2)=O)C1c1ccccc1 C(C(C)N=c1[nH]n(C)c(C(F)(F)F)c1[N+](=O)[O-])N(C(CCCCC#C)=O)C Cc1c(C(=O)N2c3cnn(c3)C2)cnn1C.c1(SC2CCNCC2)ccccc1 c1(C(=O)NCC2N(C(C3CC(C)C3)=O)CCCC2(C)C)ccc2ccccc2n1 N1(C(C(C)N(C(C)C(F)F)C=O)C)CCN(c2ccccc2)CC1 N1(C(c2oc(C)c(CO)c2)=O)CC2(CC(NC(=O)CCOC3CCCOC3)C2)C1 c1(C2(C(=O)NC(C)CC3CCN(C(=O)CO)C3)CCC2)ccc(Cl)cc1 C(=O)(CCC(=O)NN(C)C)NC(C)CNC(=O)CC1CCSCC1 c1(SC)ccc2cc(C(=O)NC34CCC(C3)N(C(C3CCSC3)=O)C4)[nH]c2c1 N1(C(C(C)OCC#C)=O)CCCC(O)(CNC(c2ccccc2C2CC2)=O)C1 CCCC(C(=O)NCCCN(C(=O)C(=Cc1cnn(C)c1)C)C(C)C)NC(N)=O C1(C(C)NC(=O)CCCN(C)C)CCCN(C(c2cnc(N3CCCC3)s2)=O)C1 c1(C(=O)NC2(CC(=O)NC3CC(=C)C3)CCC2)c[nH]nc1C C1(C)(C(=O)NCC2(C)CCN(C(CCC3CC(OC)C3)=O)C2)CCC(F)(F)C1 c1(C(=O)NC2CCC(NC(c3n(C)ccn3)=O)C2)ccc(Br)c(Cl)c1F C1(C(=O)NC(C)C(C)(C)C)CNC(=O)C12CCN(C(=O)Cc1ccccc1)CC2 N1(C(C=CCCC)=O)CCCCC1C1(CNC(=O)CC2OCCO2)CCOCC1 c1(OC)ccccc1C(=O)NCC(=O)NCC#CCNC(C1(F)CC=CCC1)=O c1(NC(C(C2CCCCC2)OC)=O)cc(O)ncn1.C12CC(F)(C1)CNC2=O N1(Cc2cccc3c2CC(C)(C)C3)CCC12CCC(F)(F)CC2 CC1(C)CCN(C(=O)CC2CC(OC(C)(C)C)C2)CC1NC(C1CCC(F)(F)C1)=O C1(NC(C(COC)(C)C)=O)CC2CC1CN(C(=O)CCCCc1ccccc1)C2 c1(CNC(=O)CCc2cc(Cl)cc(Cl)c2)ccc(S(=O)(=O)NCCO)s1 CCCC(C)(CC)C(=O)N(CC(CC)NC(=O)Cc1cccc(C)c1)C C123C4C5C1C1C2C4C51C(=O)NC(C)C1CN(C1)C3=O.c1(C(N)=O)c[nH]c(C(N)=O)c1 CCCCCC(F)C(=O)NC(C)C(=O)N(CC(O)C1CC1)C C(=O)(CS(=O)(=O)c1ccccc1F)NC1CCN(C(C2CC(C)(O)C2)=O)CC1F c1(OC)cc(C)c(C(=O)NCC(C)(C(C)(C)C)NC(=O)COC2CCOC2)cn1 CC(C(=O)N1CCOC(CCNC(=O)CCSCC(N)=O)C1)C(F)(F)F c1(CC)cccc(OCCC2CC2)c1.C1(C(=O)OC(C)(C)C)CC2CC2N1 C(C(C)C(F)C(=O)NCc1ncc(CC)s1)NC(c1n(CCC)ccc1)=O C(CC1(C)CCOC1)(C(=O)NCC(F)F)N1CCC(CC(=O)OCC(C)C)C1 c1(C(N2CC(CNC(CC3(C)CCCO3)=O)OCC2)=O)ccccc1[N+](=O)[O-] c1(C(=O)NC2CCC(C(=O)NCC3CCO3)C2)cccc(-c2ccncc2)c1 Cc1cc(NC2CS(=O)(=O)CC2C)ncc1S(=O)(=O)N1CCC(NC(C)C)CC1 C(=O)(CCC(C)S(C)(=O)=O)N.C(=O)(CCS(C)=O)N(CCCNC(COC)=O)C c1(C(=O)NC(C2CCOC2)CNC(c2c(OC)ccs2)=O)cccnc1OC c1(C(=O)NCC(C)N(CC)CC)ccc(=O)n(CCSc2ccc(Cl)cc2)n1 C=CC(CC)C(=O)NC(c1nc(=O)o[nH]1)C N1(C(C(C)(C)O)=O)CCCC2(CNC(=O)CCF)CCCC12 C12(NC(c3nc(C)[nH]c3C(F)(F)F)=O)CCC(C1)N(C(C1(O)COC1)=O)C2 C1(NC(c2ccc(COC)[nH]2)=O)CCN(C(c2ccoc2C(F)(F)F)=O)CC1O c1(CCC)cc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)C2C)sc1C CC(CC(=O)N1CCN(CCC2CN(C(=O)OC(C)(C)C)C2)CC1)C(F)(F)F CC(CC=CCl)(C(=O)NCC1(NC(C2CCC(=O)C2)=O)CCC1)c1ccccc1 C(c1ccc(F)c(F)c1)=C(C)C(=O)NCC(CO)NC(=O)C(C)C(O)C(C)C CC1CCC(N=c2[nH]c(=NCc3cccc(C(C)(F)F)c3)[nH]c3c2COC3)CC1 Cc1ccc(C(=O)NC2CC3CC(NC(C4CCCS4)=O)C2C3)c(C2CC2)c1 c1(CCC)ccc(OC(=O)CC2(OC)CCOC2)cc1.SCC c1(CNC(C2CCS(=O)(=O)C2)=O)nc2c(s1)CCN(C(=O)C(O)CC1CC1)C2 CC(C(F)C(=O)NCCCOCCNC(c1cn2ccnc2s1)=O)C(F)(F)F Cc1cc(C(=O)NCC2CC2NC(=O)C(C)(F)c2ccccc2)cs1 C1(CC(=O)N(CC)Cc2ccoc2)C2CN(C(C3(C(=O)OC)CC3)=O)CC12 C(CCCC(=O)NCC(c1ccccc1F)NC(C1CCC(F)CC1)=O)N(C)C N1(C(C(c2cc(CO)no2)C)=O)CC2(CC(CNC(=O)CC(C)C3CCCO3)C2)C1 c1(CCC(=O)NCCCN(C(=O)C(O)CN(C)C)CC)ccccc1 N1(C(CCSCCC)=O)CC=C(CC(=O)NCc2coc(C)n2)CC1 C#CC1CCN(C(C2CCC(CNC(=O)CCCCN(C)C)C2)=O)C1 CN1C(=O)CCC1CC(=O)NC(Cc1cn(CCCCCN(C)C)nn1)C(=O)O C1(C(N2CC(F)(C(=O)NCCC(C)N3CCC3)C2)=O)CC(C)N(C)C1 CN(C(=NCCc1ccc(Cl)cc1Cl)NCC(O)CF)Cc1ccnn1C Cn1ccc(=NC(=O)C(=O)NCc2ccc(CN)cc2)[nH]1 N1(C(=O)CN2CC3CC3C2)CC(Nc2ncnc3ccsc23)C2(CCOCC2)C1 C(CN=c1nc2[nH][nH]cc-2c(O)n1)(C1CC1)NC(C1CCC2(CC2)C1)=O Cc1ccc(C(=O)NC(C2CCN(C(=O)CSCc3ccc(Cl)s3)C2)C)nc1 C12(NC(C(CC)CC)=O)CC(CO)(C1)OC21CN(C(=O)C(C)C2CCCC2)C1 c1(C(N2CCN(C(C=C=C(C)C)=O)C(C)C2)=O)ccc(P(C)(C)=O)o1 N1(C(C2C(C(C)O)C2)=O)CC(CNC(=O)C(C)(C)C2CCCCC2)OC(C)(C)C1 C(=O)(CCCc1ccsc1)NCC(C)(C)C(CN(C(C)=O)CC)CO C(=O)(C(N=[N+]=[N-])C(C)C)NC(CNC(CC=CC)=O)COC C(C(C)CN(C(=O)CC1CCOC1)C)OC.C12CC(C1)NC(=O)C2 CCC(C)C(O)CC(=O)N1CC(O)(C(F)C(=O)Nc2c(C)csc2C)C1 c1(C(N2CC(O)(CN(C(C3=C(C)OCC3)=O)C)C2)=O)cc2c(nn1)CCC2 C1(CN(C(C2(CCC=C)CC2)=O)C)CCCN(C(c2nn(C)cc2N)=O)C1 c1(C(N2C(CNC(c3cc4sc(Cl)cc4[nH]3)=O)C=CC2)=O)cn2c(n1)CCCC2 O=C(C1=NOC2(CCC2)C1)NC1CN(C(c2ccoc2)=O)CC2CC12 c1(CC)ccccc1CC(=O)NC1(CF)CN(C(c2n[nH]c(C)c2C)=O)C1 c1(NCC2CN(C(Cc3c(CC)cccc3)=O)C2)ccc(C#N)nn1 C1(NC(C)Cc2cccc(N(C)C)c2)C2CC1N(C(=O)C=CC(=O)O)C2 c1(C(=O)NC2CCCN(C(C3C(CC)N(C)CC3)=O)C2)cc(F)cc(OC)c1N C(C)(N=c1ccnc(Cl)[nH]1)C1CCN(C(CCC(=C)Br)=O)C1 N#CC1(NC(=O)CSC(C)=O)CCN(Cc2cccc(C(F)(F)F)c2)C1 CC1(NC(c2cc(C3CC3)nc(O)c2)=O)CCCN(C(C2CC3CC2CO3)=O)C1 C(C(N=c1[nH]ncs1)C1CCC1)NC(=O)C=Cc1cccnc1 N1(C(CCC(=O)OC)=O)CCOCC(C)(CNC(C2COCCC2(F)F)=O)C1 N1(C(c2cc(OC)ncc2)=O)CC2CC1CN(C(c1ccc3c[nH]nc3c1)=O)C2 Cc1nn(C)c(C)c1C(=O)NC1COC2(CNC(=O)CCCC#N)CC1C2 C1(CC(=O)Nc2cccc(-n3cnnn3)c2)CN(C(=O)CSC(F)(F)F)CC1O CC1(C)CC(C)(CNC(=O)CC2CN3CCC2CC3)CN1C(c1ccon1)=O c1(C(=O)NCC(CN(C(=O)CC2C=CCCC2)C)(C)C)ccc(-c2cc[nH]n2)s1 CC1CCCC(C)N1CCC(=O)NCC(C)(C)NC(C1(C2CCCO2)CCC1)=O c1(CC(=O)NCCCCNC(=O)CC2CC(=O)NC2=O)ccnnc1O c12cccc(c1)-c1nc(C3CCCO3)nn1CC2.C(CC(F)(F)F)OC c1(CC)nc(CC(=O)NCC2CC(F)(CNC(C3C4CCCC34)=O)C2)cs1 c1(C(=O)NCCN(C2CCCCC2)C(CC2CC(=C)C2)=O)cc2ccc(F)cc2s1 C(=O)(C(CC)C(F)(F)F)N(CCC)CCNC(=O)C(c1nc(F)ccc1Cl)C C12(CNC(c3ccc(C)c(O)n3)=O)CCCC1CCN2C(=O)CC=C(Cl)Cl C1(CNC(c2cccc(C)n2)=O)CN(C(c2ccn(C)c2C2CCC2)=O)CCCO1 Cn1ncc2c(C(=O)NC3CCCN(C(C4(C)C=CCC4)=O)CC3)cccc12 c1(CC(=O)NC(CNC(c2n[nH]cc2Cl)=O)C2CC2)cnnn1-c1ccccc1 CCC(CC)(CCOC)C(=O)NCCCN(C(=O)CCCC(N)=O)C1CC1 c1(C(N(CCC(C)NC(C2(C#C)CCC2)=O)C)=O)n[nH]c2ccc(F)cc12 C(C)(CCC#N)(c1n(C(CC)C)nnn1)NC(c1sccc1Cl)C N1(C(C2(OC)CCC2)=O)CCC(C2(CNC(=O)CCC(C)C)CC2)CC1 c1(CNC(NCC2COC(=O)O2)=NCC2CCC2)ccc(Br)cc1Cl N1(C(CC2CCC(C)O2)=O)CC2CCN(C(C3CCOCC3(C)C)=O)CCC2C1 c1(CSc2n(-c3c(CC)cc(F)c(F)c3)nnn2)cc2ccccc2o1 C1(OC)CCC(CCNC(=O)NCc2ncn(C3CC3)n2)CC1 c1(C(=O)NCCOC2CN(C(C(C(C)O)N)=O)C2)n[nH]c2c1COCC2.C(N)(=O)N N(C(=NCCN1CCCC1)NCc1ccc(CO)o1)CC1CCCC(N(C)C)C1 c1(C(=O)NCC2(CNC(CC3C(OC)C3)=O)CCC2)cc(C)cc(Br)c1 Cc1ccc(C(=O)NCC2(C(N3CCCC3CC3CC3)=O)CCC2)nc1C n1(CC(=O)NCC(C)N(C(c2onc(C)n2)=O)C)c(C)ccc1C C(C(C)C(=O)N(C(C)C(=O)NC(C)CCN(C)C)C)OC(C)=O C1(O)(CN(C(c2c(COC)scc2)=O)C)CCN(C(C2CC2(C)C)=O)C1 c1(C(N(C2CCCC(NC(=O)CN(C)CCO)C2)C)=O)cccc2oc(=N)[nH]c12 C(=O)(C1CCSc2ccccc21)N1CC2N(C(c3cc(OC)ns3)=O)CC(C2)C1 N1(C(CCC(C)OCC)=O)CCC2CN(C(=O)C(C)=CCO)C2C1 C(=O)(CC(C)C(=O)NCC1(NC(c2coc(C3CCCCC3)n2)=O)CCC1)OC c1(N(S(C)(=O)=O)C(C)=O)ccc(C(N2CCC(NC3CCCC3)CC2)=O)cn1 N1(CC(=O)NC2CC2)CCc2cccc(CNC(c3ccncn3)=O)c2C1 N1(C(C=Cc2cn(C)nc2)=O)CCOCCC1C(=O)NCC1C2CCCCC12 C(=O)(C(O)C(C)(C)C)NCC(CC)NC(c1ccc(Br)cc1)=O c1(C(N2CC(CNC(c3c(C)ncc(N)c3)=O)C(O)C2)=O)c(C)cc(Cl)cc1C c1(C(N(C2CN(C(c3cn(C)nc3Cl)=O)C2)C)=O)ccc(-c2ccco2)cc1F c1(C(=O)NC2CC(C)(CNC(c3cnc(OCC)s3)=O)C2)cc(F)c(N)cc1F C(=O)(CC(C)C(C)C)NC(CCN(C(C1CC(=C)C1)=O)C)C(C)C c1(CNC(c2cn(CC3CNCCO3)nn2)=O)ccc2c[nH]nc2c1 N1(Cc2ccc(C(C)=O)s2)CC(C)Sc2ccccc21 CCCCCCCCCC(C(=O)NC(C)C1CC1)N1CCC(n2ccnc2)CC1 C1(C(=O)NCC2C(NC(Cc3cccc(C)c3)=O)CC2)CC(=O)OC1(C)C c1(C(=O)NC)cccc(C(C)NCC(Cc2cccnc2)CN)c1 c1(OC)ccc(C)cc1C=CCNC(=O)NCC12CCCC1OCC2 C1(C)(CCNC(CC2(COC)CC2)=O)CCCC1.C1(C2CCOC2)C(=O)N1 C1(C(=O)NCC(CC=C)(C)C)CN(C(=O)CC2(NC(C)=O)CC2)CC(C)O1 c1(C(=O)NC2CCC(NC(C3(COC)CCC3)=O)C2)cn2c(n1)CCC2 c1(-c2cn(CCC(C)(C)NC(C3(C)CCC3)=O)nn2)cccc(CO)c1 N1(C(c2cnc(OC)nc2)=O)CCC(NC(c2cnc3n2CCS3)=O)C(C)(C)C1 C=CC(CCC)CC(=O)NC(CC(C)CC)C(=O)Nc1ccc(Cl)cc1 CCCCC(CNC(c1nnc(S)n1C)=O)NC(=O)COC1CC(F)(F)C1 c1(CC)cc(=NCC2(F)CC(NC(=O)CN3CC4CC4C3)C2)[nH]c(CC)n1 C1(C2(O)CCOC2)(C(N2CCC(CNC(CC)=O)C2)=O)CC1 C1(NC(C(C)C#N)=O)CN(C(c2cnn3cccc(Cl)c23)=O)CCC12CCC2 Cc1ccc(OCC(=O)NC2CC3(C2)CC3NC(=O)Cn2cnnc2O)cc1C C1(CNC(c2ccccc2)=O)CN(C(C2CC3CC2C3)=O)CCC1(F)F C(=O)(C(CCC(C)C)NC(c1cnncc1OC)=O)N1CCC=C(C)C1 c1(OCC)ccc(NC(C)CNC(=O)C(O)CCS(C)=O)cc1[N+](=O)[O-] N1(C(C(CCCCC)O)=O)CCOC2(CCCN(c3cnc(C#N)c(C#N)n3)C2)C1 c1(C(=O)Oc2ccc(C(=O)OC)cc2C2CC2)cc2cc(F)ccc2cn1 C1(CC(=O)OCC)CCC(C)N(C(C2CCC(NCCN3CCC(C)CC3)C2)=O)C1 c1(C(N2CCC(O)(CC(=O)NCc3cccnc3)CC2)=O)ccc2c(c1)CCO2 C1(NC(c2cc(CNC(C(C(CC)C)N(C)C)=O)on2)=O)CCC2(CCC2)CC1 c1(C(N2CC(N(C(C3C(C)C3)=O)C)C3(C2)CC3)=O)c(F)cc(N)cc1F C1(NS(CC)(=O)=O)CN(Cc2cccc(O)c2)CC12CC2 c1(C2C(C(=O)NC3CCC(NC(=O)CCF)C3)C2)ccc(F)cc1F c1(CN2C3C(C(=O)Nc4ncc(F)cc4I)C(C3)C2)ccc2ccc(Br)cc2c1 n1(CC)c(N(C(C2CCCCC2)C)CC)nnc1C1CCCCN1C C(=O)(C(N)(CC(C)C)C(C)(C)C)N1CCC(N(C(C(C)C)=O)C)C1 n1(CCOCC)cc(C2(C)CN(C(c3ccoc3I)=O)C2)nn1 n1(CC)nc(C(=O)N(CCCNC(C2(c3nccs3)CC2)=O)C)cc1C1CC1 c1(C(=O)NC2CCCCN(C(CC(C)C3CC3)=O)C2)n[nH]c2ccc(Cl)cc12 c1(C(N(CCNC(=O)CC2COC(C)(C)O2)CC)=O)cc2ccccc2nc1O C1(C(N2CCC(C(C)NC(=O)CN=S(C)(C)=O)C2)=O)CCOC2(CCCCC2)C1 c1(C(=O)NC2CCC(C)(CNC(c3c(C)cc(C)o3)=O)C2)cc2cccnc2o1 C1(CC)C(NC(C2CC3(CCCO3)C2)=O)CCCN1C(c1ncc(F)cc1N)=O N1(C(Cn2ccc(C)c2)=O)CCC(C)C1C(=O)NC1CC1CN(C)C N1(C(C2(CCC=C)CCCC2)=O)CCCN(C(=O)Cc2cn(C)cn2)C(C)C1 C(C)(C(=O)NNc1ccc(NC(c2cccc(CN)c2)=O)cc1)OC C1(CNC(C(C)(C)OCCC)=O)CCCC(NC(C2CC3C=CC2C3)=O)C1 N1(C(C(C)N(C(C(CCC)F)=O)C)=O)CC2CCC(C1)C2C#N c1(NC(C2CCC(NC(C(CCC)OC)=O)C2)=O)cc(C)c(F)cc1O CN1CCc2ccc(C(N3CCCC3CNC(C3(C)CCC(=O)NC3)=O)=O)cc21 C(=O)(CCCCC(F)(F)F)NCC(CC(C)C)NC(=O)CCc1cccnc1Cl c1(CC)nncn1NC(=O)CCN(C(=O)C=C(C)C(F)F)C(C)C C1(NC(C2CN(C)C(=O)N2)=O)CCS(=O)(=O)C12CN(C(=O)C1=CCCC1)C2 CCCC(CC(C)C)C(=O)N(CCCCN(C)C(c1nc(C(C)C)oc1C)=O)C C1(C(N(C2CCC(C(N)=O)C2)C)=O)CCN(C(=O)CCCCC2CC2)CCO1 C(=O)(C(C(C)C)C1CCC1)NCC1(CNC(c2cn(CCOC)nn2)=O)CCC1 C1(S(N)(=O)=O)(C(=O)NC2C(NC(C3(C)CCC3)=O)COCC2)CCC1 C12(NCc3cccc(OCC#N)c3)CC3CC1C2C3C(=O)OC C(=O)(CC(C(F)F)C1CC1)NC(C)CN(C)C(C1(Cl)CC1)=O c1(C(N2CCC(N(C(C3C(=C)CC3)=O)CCO)CC2)=O)cc(O)cc(Br)c1 C1(CNC(c2c(C)coc2)=O)CC2CCC1N(C(C1(C)CC1Br)=O)C2 C(=O)(CCCCC(N)=O)NCC1CCC(NC(c2n(CC)ncn2)=O)CC1 C=CCC(CC=C)C(=O)NC1CCN(C(c2coc(C)c2)=O)C(C2CC2)C1 Cc1ccc(CCC(=O)N(c2cc(Br)ccc2Cl)C)cc1F C(=O)(C1CSc2ccccc21)NC(CNC(c1c(C(C)C)scn1)=O)CO CC1(C)CN(C(=O)CSc2nncs2)CC1NC(=O)C(F)C(F)(F)F c1(CC(=O)NC23CC(C(=O)NC(C#C)C)(C2)C3)cccc(C)c1 N1(C(Cn2c(C)ncc2)=O)CC(CNC(C2CC2C(C)(C)O)=O)C2(CC2)C1 C1(CC(=O)N(CCCNC(=O)CC(C)O)C(C)C)CCCC1(F)F c1(N(C2(C(=O)NC(C)CCNC(C3CC3(F)Cl)=O)CC2)CCO)ccccc1 c1(C(N(C(C)CNC(=O)C(F)C(F)(F)F)C)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(c2cc(C)ncc2C)=O)CC23CCCC2(C1)CN(C(=O)Cc1cnns1)C3 C(CC1CC1)(CN=c1[nH]c(N2CCc3c(nnn3C)C2)nc2c1COC2)OC c12cc(oc1C)C(=O)NC2=O.C1(NS(C)(=O)=O)CCCC1CN Cc1cnnc(C)c1C(N1CCC(C(F)C(=O)N(C)CC2CCCC2)C1)=O C(=O)(CCCCCCNC(c1cc2ncccc2[nH]1)=O)N1C(C)(C(=O)OC)CC1 C(CC(=O)NC1COCC1CO)(C(F)(F)F)NC(c1ccc(=N)[nH]n1)=O C1(NC(=O)C#CC2CC2)CC2(CCN(C(c3ccc(CC(N)=O)cc3)=O)CC2)C1 N1(C(C(c2ccc(F)c(F)c2)C)=O)CCC(C)C(NC(=O)CCc2ccsc2)C1 c1(NC(C2C(CNC(c3ccn(CCOC)n3)=O)OCC2)=O)c(O)cccc1F N1(C(C=CC(C)(C)SC)=O)CCC2(C1)CN(C(c1cn3ccsc3n1)=O)CCO2 Cc1c(CC(=O)NC(C(=O)N(C(CO)C2CC2)C)C2(O)CCC2)ncn1C N1(C(c2ccc(C)o2)=O)CCCC(NC(C2(NC(C)C)CC2)=O)C(F)C1 C12(C(=O)NC3C(C)C3(C)C)CCCC1CN(C(=O)CC13CCCC1C3)C2 C1(NC(CNC(=O)OCC)=O)CCN(C(C2CCC(F)C2)=O)CCC1CO C(=O)(C(C)CS(C)(=O)=O)N1CCN(C(Cc2cc(C)sc2)=O)CC1CCO N1(C(CNC(CC)=O)=O)CC(C)(C)C(NC(c2ccncc2NC)=O)C(C)(C)C1 C1(C(=O)NC(CC)CN(C)C(c2cnn(CC(F)F)n2)=O)(CC)CCCCC1 CC(C)(C(=O)NCC(=O)NCc1ncoc1C1CCCO1)c1ccno1 CS(=O)(=O)C1(C(=O)NC(CNC(c2ocnc2C(F)(F)F)=O)C2CC2)CCCC1 c1(-c2ccc(C(=O)NCc3cnc(C)s3)cn2)cc(O)cc(F)c1 c1(C(=O)NC2CCC(CNC(CC(C=C)C)=O)CC2)cnc(C(F)F)cc1C C=C(C)CC(C)C(=O)NCC1CN(c2nnc(-c3ccccc3)s2)CCO1 C(=O)(C1=CCC(C)(C)CC1)N1CC2C(NC(CCCOCC=C)=O)CC(C2)C1 c1(C(=O)NCCC(=O)NCCC2N(C(COC)=O)CCCC2)cc(N)nc(Cl)c1 N1(C(c2c(C)noc2)=O)CCN(C(=O)C(C)NC(c2ccco2)=O)C2CCC12 c1(C(N2CC3C(CN(C(C=CC=CCC)=O)CC)C3C2)=O)nccn2ccnc12 c1(C(N2C(C)CC(NC(c3cnc(Cl)c(N)c3)=O)C2)=O)ccc(C2CC2)cc1F c1(C(c2n(CCOC)nnn2)NCc2ccncc2Br)cccc(Cl)c1Br C1(C(N2CCOC(C(=O)NCCCP(C)(C)=O)C2)=O)(CC)CCNC1=O C1(C(N2CC(C(=O)NC)C2)=O)CCC(C(C)C)N1C(=O)Cc1cccc(F)c1 C(CO)(C(=O)N1CCC(CNC(=O)C(C2CC2)N(C)C)C1)N(C)C C1(CC)CC(C)CN(C(=O)C(C)(CO)NC(C2CC(=O)C2)=O)C1 c1(C(=O)NCCCCNC(C2(F)CCC(C)CC2)=O)ccc2c(c1)OC(C)(C)C2 N1(C(c2n(CCC)ncc2)=O)CCCCC1CCC(=O)NCC1CCC(F)(F)C1 N1(CC)CC(C(=O)NC2CC(CNC(=O)CCCCC3CC3)C2)CCC1=O CC1(C)CC(NC(C2CCC(CO)CC2)=O)CN1C(=O)CCCCCF c1(C(N2C(C)CC(CNC(Cc3c(C)nc[nH]3)=O)C2)=O)cccn2[nH]c(=N)nc12 C1(NC(C(CC)OCC)=O)CCN(C(C2CC2CN(C)C)=O)CC1F CC(C)CC(C(N)=O)N(C)C(C1CCCCN1C(=O)CCC(C)C)=O N1(C(CCCC#C)=O)CCCC2(CCN(C(=O)C(C)(O)CCc3ccccc3)C2)C1 Cc1cc([N+](=O)[O-])ccc1C(C)NC(c1ccc(Br)c(Cl)c1)C C1(CC#C)(C(=O)NCC#CC(=O)OC)CCN(C(c2ccncc2CC)=O)C1 C12(C(=O)NC3CN(C(c4c(C)nc(C(C)C)s4)=O)C3)CCCC(C)(C1)OC2 N1(C(C(CC)N(CC)Cc2ccco2)=O)CCN(c2ccccc2C)CC1 C1(C(=O)NCC2(C(=O)NCc3ncc(C)o3)CCCO2)CC(F)C(=O)N1 C1(F)(C(=O)NC2CCN(C(c3c(C)cccn3)=O)CC2O)CCCCC1(F)F c1(NC2N(c3cc(NCC(CN(C)C)O)ncn3)CC(O)C2)ccc(Cl)cc1Cl n1(-c2ncc(C(=O)NCC(C)NC(c3c(C)scc3)=O)s2)cnc2ccccc12 O=C1CCN(CCC2CCC=CCC2)C(=O)N1CCOCC1CCCC1 Cc1c(NCCCN2CCOC2=O)ncnc1NC(c1ccncn1)C c1(C(=O)NC(CCNC(Cc2cc(OC)c(Cl)cc2)=O)C)cccc2oncc12 C1(C(=O)NC2CCC(COC)C2)CC2(CCN(C(=O)CN=[N+]=[N-])C2)C1 Cc1ccc(C=CC(=O)NC2CCN(C(=O)C(C)C3CC3)C2C2CC2)o1 c1(C(N2CC3C(NC(CC(C)C4CC4)=O)(C3)C2)=O)ccc(F)c(O)c1 c1(C(=O)NCC2N(C(CC#N)=O)CC2)cc(=O)c2ccc(Br)cc2o1 N1(C(C(c2cn(C)nn2)NC(C=C(C)C)=O)=O)CCc2ccncc2C1 c1(C(N2C3CN(C(CSC(C)(C)C)=O)CC2CC3)=O)ccc2n[nH]cc2c1Cl C1(NC(c2ccc(SC)cc2C)=O)C2CCC1CN(C(=O)CN1CCOCC1)C2 Cc1nn(C)cc1C(N1CC2C(C(=O)NCC3COCCO3)C2C1)=O c12ccc(o1)C(=O)N(C1CC1)CC2.C(C(=O)NCC1CC1C)N(CCC)C Cc1cc(Cl)cc(C(N2CC3CCC2CN3C(C2CCC2(C)C)=O)=O)c1N c1(C(=O)NCC(CC)NC(=O)C(O)CN(C2CCCCC2)C)cccc(F)c1F O=S(=O)(c1cccnc1NCCOCF)NCC(CCO)c1ccncc1 N1(C(C2CC(CCC)C2)=O)CCC(F)(n2cc(CS(=O)(=O)CC)nn2)CC1 Cn1cc2c(n1)CC(C(=O)NCC1(NC(c3cscc3F)=O)CC1)CC2 N1(C(C2CCC(OCC)CC2)=O)CC2CC1CC2CNC(c1nonc1CC)=O C=C1C(NC(=O)NCC(c2ccc(F)cc2F)OC(C)C)CC2CC1C2(C)C C1(CC#C)(C(=O)NCC(C)(C)NC(=O)Cn2cc(CO)nn2)CCCC1 C1(C(=O)OC)COCCN1C(=O)NC1CCCOC1c1ccc(C(C)(C)C)cc1 C1(NC(CCC2C(C)(C)C2)=O)CN(C(c2csc(=N)[nH]2)=O)Cc2nccn2C1 c1(OCC)cc(C(N2CCC(NC(=O)CC3CC34CC4)C2)=O)cc(Cl)c1O n1(CC)cc(C(=O)NC2(C3CCCN3C(=O)C(C)(C)Br)CC2)cn1 c1(C(=O)NC(CC)CNC(=O)C(CO)NC(N)=O)ccc(O)c(C)c1C CCS(=O)(=O)c1ccccc1CC(=O)NC(CNC(C1CC1[N+](=O)[O-])=O)C(C)C N1(C(=O)OC(C)(C)C)CC2CC(C1)C2NC(=O)Cn1nnnc1-c1ccsc1 c1(OC)ncc(C(=O)NC2(CC(=O)NCC3CNC(=O)O3)CCC2)cn1 C1(F)(C(=O)NC(C)(CNC(=O)COC(F)F)C2CC2)CCOCC1 C1(c2cn(C)nc2)CN(C(=O)C=CC(C)(C)C)CCN1C(=O)CC1CCCCC1 c1(C(=O)NC2CCCCN(C(CC(CCC)C)=O)C2)cccc2c(O)nncc12 c1(CC(N2CC(C(C)NC(C(C)O)=O)C2)=O)nc(F)c(F)cc1F C(=O)(C(C)(C)C)N(CC(CC)NC(c1coc(C2CCCCC2)n1)=O)C N1(C(C2CC(=C)C2)=O)CC=C(CCNC(c2cncc(C(F)(F)F)n2)=O)CC1 C1(CNC(C(CSC)(C)NC(c2sncc2C)=O)=O)CC(O)C12CCC2 C1(NC(c2c(C)n(CCO)nc2)=O)CCCCN(C(=O)C(C)(C)c2ccns2)C1 N1(C(C2C(CC)N(C(c3ccnc(C)n3)=O)CCC2)=O)CCC(O)C(F)(F)C1 C1(C(=O)NCCCCCNC(c2cnc(OC)nc2C)=O)CCc2nc[nH]c2C1 c1(C(N(C)CC2CCN(C(C3CC(C)(C)O3)=O)C2)=O)nnc2n1CCCCC2 N1(C(C(CC)O)=O)CC(CNC(c2cnc(C)nc2C)=O)CC1(C)C c1(C(=O)NC2CC(CCNC(COCC(=C)C)=O)C2)cccc(Cl)c1[N+](=O)[O-] C1(C(=O)NCc2cn(CC(=O)N(CC(N)=O)C)nn2)CCCCC(=O)C1 C1(O)(CNC(=O)CCn2cc(Cl)cn2)CCN(C(c2cnn(C(F)F)c2)=O)CC1 C1(C(=O)NCCSC)CN(CC(=O)Nc2ccccc2C)C2(CCC2)C1 c1(OC)ccc(CC(=O)NC23CCC(C2)N(C(C2CC2C)=O)C3)c(F)c1 CCC(CC)C(C)C(=O)NC1CC(NC(c2cc(F)cc(F)c2)=O)C(O)C1 c1(C(=O)NC(CC=C)CNC(=O)CCOCC)cn2ccc(C)cc2n1 CCCCCCC(F)C(=O)N1CCCC1CNC(c1cnnc(C)c1)=O c1(C(=O)NCC2N(C(C(c3ccc(C)cc3)C(C)C)=O)CC2)ccc(C#N)cn1 C1(NC(Cc2c(C)noc2)=O)CN(C(=O)C=CS(C)=O)CC(C)(C)C1 c1(OC)c(CC(N2CC3CC2CC3NC(=O)CCC2CCC2)=O)cccc1F CC1CCN(C(c2cc(CNC(=O)C=CC(F)(F)F)cs2)=O)CC1O Cc1ccc(NC(N2CCC(C)(NC(=O)Nc3ccccc3)C2)=O)c(S(C)(=O)=O)c1 C1(C(N(C2CCCCCC2)CCNC(C(C)OCC#C)=O)=O)CC2C=CC1C2 c1(SCC(=O)NC(CC(C)NC(C2(C#C)CCC2)=O)C)ccc(C)cc1 C1(NC(=O)C(F)=C2CCC2)CCN(C(c2scnc2C2CC2)=O)CC1CO N1(C(c2c(OCC)ccs2)=O)CC(NC(=O)C#CC(=O)N(C)C)CC12CCOC2 CC(=Cn1ccnn1)C(=O)N1CCC(C)(C)C(NC(C2Cc3nncn3C2)=O)C1 C(=O)(C(C)(COC)CC)N1CCCC(NC(C(C)=C(CC)C)=O)C1 c1(C(=O)NC(C)C(=O)C2CC2)nccc2c(Cl)cccc12 c1(NC(C(CO)NC(c2ccn(C)c(=O)c2)=O)=O)ccc2cnccc2c1 C1(CCC)(C(N2CCC(O)(CNC(c3ncsc3C)=O)C2)=O)CCNC1=O c1(C(=O)NCCC(C)N(C(=O)COCC2CCOC2)C)cccc2ccoc12 c1(CC)cc(F)ccc1NC1(CC)CC(c2nnnn2CC2CCCO2)(OC)C1 c1(C(=O)NC2CN(C(c3nsnc3O)=O)C2)cccn(CC(=O)NC2CC2)c1=O CC1(C)CCC2(CC1)CC2C(=O)NCCOc1ccccc1C#N CCCCC(CC)CCC(=O)N(CCNC(=O)CC1CCCCC1F)CC c1(C(=O)NCC2CC(Nc3nc(O)n(C)c(=O)c3)C2)noc2c1COCC2 C(=O)(CCC(=O)N1CCC(C)(CNC(C2(c3cccc(Cl)c3)CCC2)=O)C1)NC c1(SC(C)C(=O)NCC2CCN2C(=O)C(O)Cc2ccccc2)nncn1C C=C=CC(C)C(=O)NC1(c2ccccc2)CC(NC(=O)C(C)CC2CCCC2)C1 NS(=O)(=O)CCCC(=O)N1CCCC1C1(NC(C23CSC(C2)C3)=O)CC1 N1(C(C2(COCC)CC2)=O)CCC(F)C(NC(=O)Cc2ccc(C)cc2C)C1 c1(C(N(C)CC)=O)nnc2ccccn12.C1(OCCCC)CC(CO)C1(C)C C#CCC(C)(C)C(=O)NCC(N1CCN(C(C2CCCSC2C)=O)CC1)C c1(SCC#C)cccc(C(N2CCC(CN(C(=O)CCC3OCCO3)C)C2)=O)c1 Cc1cc(CN2CC(NC(=O)NC(=O)NCCCl)C2)c(I)cc1F C(CCC(C)(C)NC(c1cnc(O)n1C)=O)NC(C(N1CCCCC1=O)C)=O Nc1cc(Cl)ccc1C(N1CCN(C(c2csc(SC3CC3)n2)=O)C2CC12)=O c1(NC(=O)Nc2c(CC(C)C)cccc2)cc(CO)c2c(c1)OC(F)(F)O2 c1(OC)ccc2[nH]c(=NC(C)C3CCCN(C(C4(F)CCOC4C)=O)C3)sc2n1 c1(CN2CC(NC(C(C)OCC=C)=O)C(F)C2)ccc(C=CC(=O)O)cc1 Cc1ccc(O)cc1C(=O)NCCCCCCN(C)C(c1cnns1)=O Cc1nn(C)cc1C(=O)NCC1CCN1C(c1csc(N2CCCCC2)n1)=O C(Cc1ccccc1)(C(O)C(F)F)NC(=O)Cc1ccc(F)cn1 N1(C(C(CC#C)O)=O)CCN(C(c2cccc(Br)c2)=O)C(c2ccncc2)C1 N1(C(c2cc(C)n(C)c2)=O)CCC2CCN(C(C3(C)CCCCCC3)=O)CC2C1 C(=O)(CCCC(=O)NCCN(C(=O)CS(N)(=O)=O)C1CCOC1)OC CC(N=c1[nH]c2c(c(=NC3CCC(C)(C)C3)[nH]1)COCC2)c1ccc(Br)s1 C(=O)(C1CCCc2scnc21)NCC(C)CNC(=O)CCc1cccn1C C12CCC(O1)CCCO2.C1(C)(CC(=O)OC(C)(C)C)OCCO1 N1(C(C=Cc2c(C)nccc2)=O)CC2(CCCC2NC(c2nc(=N)cc[nH]2)=O)C1 c1(C(=O)NC(C(C)NC(Cc2c(C)n(C)cn2)=O)(C)C)ccn2cccc2c1 c1(C(=O)NCCCCCN(C(c2[nH]cc(CC)n2)=O)C)ccc(C)nc1C1CC1 c1(OC)ccccc1CCC(C(=O)NC1CCC1N1CCOCC1)OC N1(C(CN2CC(CC)C2)=O)CCC(O)(CNC(=O)CC2CCC(C)CC2)C1 N1(C(C(C)=C2CCCC2)=O)CC2(CCC2)CC1CNC(C12CC1C2)=O N1(C(C(CC=C)(F)F)=O)CCC(CNC(c2ccc(Br)cc2C)=O)C(F)(F)C1 N1(C(c2ccn(CC)n2)=O)CCC(CNC(=O)C(C)NC(C2CCC2)=O)(OC)C1 CSC1=C(C(=O)N2CCN(C(=O)C(C3CCOCC3)O)C(CF)C2)CCCC1 c1(C(N(C2CCN(C(=O)C3=NNC(=O)C3)CC2)CC#C)=O)cc(Cl)c(C)cn1 c1(NC(CCCCC#C)=O)cnn(CCNC(=O)COC2CC2)c1.C(CCC(C)C)O N1(C(C(CC=C)(C)C)=O)CC2CCCC(NC(=O)C3CCc4c[nH]nc43)C2C1 C(=O)(C(C(=O)N1CCC2(NC(c3c[nH]nc3CC)=O)CCCC12)C(C)C)OCC CN1CCC(n2cc(C3CCN(C(C4CCC4C(C)(C)C)=O)CC3)nn2)C1=O C12(NC(CC(c3ccccc3F)C)=O)CCCN(C(c3ccon3)=O)CC1C2 CN1CCc2cc(C(=O)NCC(C)(C)CNC(C3CC(C(N)=O)C3)=O)ccc2C1 CCCCCCN1CCC1.C12C=CC(C1)NC(=O)CN2 c1(OC)ncnc(C)c1C(N1CCC2(CC2NC(=O)CC2CCCC2C)C1)=O N1(C(Cc2c(O)ccc(C)c2)=O)CCC2(CCN(Cc3cc(I)ccc3Br)C2)C1 c1(NC(N2CCN(S(=O)(=O)C3CCCCC3)C3CC23)=O)cc([N+](=O)[O-])ccn1 CCC1=C(C(=O)NC2(C(N3CCOC4(CCCC4)C3)=O)CC(F)C2)CCCO1 N1(CC)C2CN(C(=O)CCC=O)CC12.C(CC(=O)OC)OCCCO CN1CCC(NC2CCN(CC(O)COc3ccccc3I)C2)CC1=O C1(NC(Cc2c(C)ocn2)=O)CN(C(=O)C(C)C2CC2)C2(CCCC2)C1 N1(C(CCN(C(C)=O)C)=O)CCN(C2CCN(C(=O)C(C)n3cccc3)C2)CC1 CCCC(CCC)C(=O)N1CC2(C1)SCCC2NC(C1CCC(=O)N1C(=O)OC)=O N#Cc1cnc(NC2CCCN(CCNC(C3(C(F)(F)F)CC3)=O)C2)c(Br)c1 C(CCCCC(=O)N1CCCC(CN(C(=O)C(c2cccc(C)c2)C)C)C1)=CC CC1(C(=O)NCC2(CO)CCN(C(C3CC(C(F)(F)F)C3)=O)C2)CCC(=O)C1 C1(C(=O)NC(CCNC(C(CC)OCC)=O)C)CCc2c(Br)cccc2C1 c1(C(=O)NC(C(=O)NCc2c(C)con2)CN(C)C)cc[nH]c(=N)n1 C1(C(=O)NC2C(NC(CCCOCC=C)=O)CCC2)CCNC(=O)C1 C=CCCCC(=O)NCC1CCN1C(=O)CC12COC(CF)(C1)C2.C(C)(C)(C)NC(=O)O C#CC1(CO)CN(C(=O)COc2cccc(N(C)CC)c2)C1 C(=O)(C1=CC2(CCOC2)C1)NC1C(NC(c2c(CC#N)ccs2)=O)COCC1 C1(CC)(NC(c2csc(C)n2)=O)CCN(C(=O)C(F)n2cccn2)CC1 N1(C(C(N2CCC(C)CC2)=O)=O)CC(CNC(=O)CNc2nccs2)C2(CC2)C1 CC1COCC(C(=O)N(CCCCCNC(=O)CC2CC3(CCC3)C2)C)O1 C1(C(N2CCN(CC(=O)NCCOC3CCCC3)CC2)=O)CCC2CC1CO2 C12(CNC(C=CS(C)=O)=O)CCC(CC1)N2C(=O)CCC1CCCCC1 CCC(CO)(C(=O)NCC1CN(C(=O)C(c2cnn(C)c2)C)C(C)(C)C1)OC c1(C(=O)NCC(C)N(C(Cc2c(C)cccc2)=O)C)ccc([N+](=O)[O-])cn1 C1(NC(CCCC(C)=O)=O)CCC2(CCN(C(C34CCC(CC3F)C4)=O)C2)C1 CN1CCN(C(C23CCCC2C3)=O)CC1CNC(c1cncc(Br)c1)=O CCC(CC(F)(F)F)C(=O)NCC1CCCC1NC(=O)CSCC(N)=O c1(C(c2nc(C3CC3)no2)C)nccc(CN2CCOC2=O)n1 CC1CCN(C(C2CCCCC2)=O)CCC1N1CCCOCC1 C1(C(=O)NCC2C(Cn3cc(-c4ccn(C)n4)nn3)C2(F)F)CC2(CCC2)C1 c1(OCC)ccc(F)c(C(=O)N(CCN(C(=O)CC(F)(F)Cl)CC)CC)c1Cl C(C)(C)(CCCC(=O)NC1(C(N)=O)CC1)NC(c1cc(C(C)=O)[nH]n1)=O CCCCCCOCC(=O)OC(C)(C)C.C1CS(=O)(=O)NCCC(=O)N1 c1(NC)cc(C(=O)OC)ccc1NC(=O)C(C1(N)CCOCC1)(C)C CC(CS(C)(=O)=O)C(=O)N1CC2CC1CC2NC(c1cc2ncccc2[nH]1)=O C1(NC(=O)NC(c2ccc(Oc3ccccn3)cc2)C)CN2CCN1CC2C c1(C(N2CC(NC(CCCC#C)=O)CC3(C2)CC3)=O)c[nH]c2ccc(Br)cc12 CCCCC(C)N=c1[nH]c(=NCC(COC)S(C)(=O)=O)[nH]c2c1CC(C)CC2 c1(OC)ccc(CC(=O)NC(C)CNC(=O)C(c2ccccc2C)(F)F)cc1F C1(NC(C(C(COC)C)C)=O)CC2CC(C1)N(C(=O)CC1CSC1)C2 C1(CNC(C2(C)CC(=C)C2)=O)CN(C(C2CC(n3ccnc3)C2)=O)CCC1C Cc1nc(C2CC2)oc1C(=O)NCCC1(NC(=O)CC2CC3(CCC3)C2)CC1 c1(NC(C(=O)NCc2ccn(C(C)C)n2)=O)cccc(-c2ccno2)c1 C12(C(=O)NC3CC4CN(C(c5cccc(NC)n5)=O)C3C4)CCC(CC1)C(C)O2 c1(C(=O)NCCCCC(C)NC(C2CC=C(C)CC2)=O)ccc2oncc2c1 C(=O)(C(C(C)(C)C)N(C)C)NCCCNC(C1C(c2c(OC)cccc2)C1)=O N1(C(C2C(=C)CC2)=O)CCC(C2(NC(=O)C=C(C)C3CC3)CC2)C1 c1(CC(=O)NCC(C)NC(CSCC)=O)ccc(Cl)c(Br)c1 C(=O)(CCS(=O)(=O)CCOC)NCC(C(C)C)NC(CCCCCC=C)=O N12CC3CC(C3)(C1)C2=O.C(=O)(CC(F)(F)F)NCC1N(C(C(C)C)=O)CCC1 C(=O)(C#CC1(C)CCCO1)N1CCCC(CNC(C(C(=C)Cl)(C)C)=O)(CO)C1 N1(C(C(CC)SC)=O)CCCC2CN(C(c3cc(S(C)(=O)=O)cs3)=O)CCC12 C1(NC(Cn2c(C)cc(C)n2)=O)CCN(C(=O)CCOCC2CCCO2)C(C)C1 c1(NC(CC(C)NC(Cc2cnc(C)s2)=O)C)nccc(C(F)(F)F)n1 c1(C(N2CCC(F)(CNC(c3nc(C)sc3)=O)C2)=O)c[nH]cc(Cl)c1=O N1(C(C2N(CC)CC2)=O)CCC(C(=O)N(C)Cc2sccc2C)(CF)C1 N1(C(C(C)C2CCC2)=O)CC(NC(=O)COC2CCOC2)CC1(C)C C1(C(N2C(CCNC(c3ccnn(C)c3=O)=O)CCC2)=O)CCn2cncc2C1 N1(C(C2N(C(CCCCCC#C)=O)CCC2CC)=O)CC2(C)COCC2(C)C1 C(=O)(C1=CCCN(C(c2c(F)cc(Br)cc2Cl)=O)C1)NC(c1ccc(C)cc1)C N1(C(c2cccc(C(C)C)c2)C(=O)NC2CC(F)(F)C2)CCCC(C)(O)CC1 N1(C(C(C)SCC)=O)CC(CN(C(C2(CO)CC2)=O)CC)C2(CC2)C1 C1(CS(=O)(=O)NC)CN(CC2CCN(C(=O)OC(C)(C)C)C2)c2ccccc2O1 c1(COC(C)CCNC(C2CC(CNC(=O)Cc3nc[nH]n3)C2)=O)ccccc1 c1(NC(c2nnnn2C)(COCC)C)nccc(Cl)c1CC N1(Cc2ccc(C(=O)NCC=C)cc2)CCC2(CC1)CC(OC)CO2 C1(CN(C(c2c(CC)non2)=O)C)CCCCN1C(C1CCC2(C1)N=N2)=O N1(C(C=C(C)C(C)(C)C)=O)CCCCC1CC(=O)Nc1c[nH]ccc1=O c1(OCC2N(C(=O)OCc3ccn(-c4ccccc4)n3)CC2)ccc(F)cc1 CCCCCCCCC(F)C(=O)N1CC(NC(=O)Cn2ccccc2=O)C(F)C1 C1(NC(C2CCCCC2C(F)(F)F)=O)C2CC1N(C(C1CC=CCC1)=O)C2 c1(CC(=O)N(CCCOCCN(C(CCC#CC)=O)C)C)cccc(C)c1Cl C(=O)(CCC1=NNC(=O)CC1)NCCCN(C(=O)C(C1CCCCCC1)O)CC N1(C(c2c(F)cccc2F)=O)CCC2CCN(C(c3cscc3Cl)=O)CC2C1 C1(NC(c2cc(OC)cc(Br)c2)C)CCCC(C)(C)CC1 N1(C(C2C(C(C)O)C2)=O)CC2CN(C(=O)CCc3ccc(C(=O)OC)cc3)CC2C1 N1(CC(c2c[nH]nc2-c2ccccc2)=O)CCC2(CC1)CC2C(=O)NCC(O)CO S(=O)(=O)(c1cc(C(=O)O)ccc1Br)NC1CCCC(OC)C1 O=C(C1=CCCCC1)NC1CC1NC(C1(Cc2cccc(F)c2)CCC1)=O c1(C(=O)NC(C)C(C)NC(=O)C2=CCCOC2)cc(Cl)c(Cl)[nH]c1=N Cc1cc2ncnc(N3CCCC3C(C)(C)CNC(=O)C(C)c3ccsc3)c2[nH]1 N1(C(CCCc2n(C)cnn2)=O)CCC(NC(=O)COC2CCCC2)C12CC2 c1(N(CCN(CC)CC)CC)[nH]c(=NCc2cc(COC)on2)nc2c1cnn2C c1(C(=O)NC(CNC(C=C(CCC)CCC)=O)(C)C2CC2)cc(Cl)c(F)cc1C N1(C(c2ccc(N)c(F)c2)=O)CC2CC1CN(C(=O)C(O)Cc1cnc[nH]1)C2 Cc1ccc(C(N2CCCCC(NC(=O)C(O)c3ccco3)C2)=O)cc1N C(=O)(C#CC1CCCOC1)N1CC(CCCNC(Cc2c(C)scc2)=O)OCC1 C1(NC(c2cn(CC)nc2)=O)COC2(C1)CN(C(c1ncsc1C)=O)C2 Cc1nn(CC(=O)NC(C)CC(C)NC(C2(C)COC2)=O)c(C)c1[N+](=O)[O-] c1(C(=O)NCC(CO)NC=O)c2c(cc3c1CCC3)CCC2.C=CCC C(C)(CCCC(=O)N1CCc2c(n[nH]c2C)C1)NC(COCCCC#C)=O c1(OC)c(C(N2CCN(CCN(C)C(C3(C)CC3(F)Cl)=O)CC2)=O)c(C)nn1C C12(NC(Cc3cc(C)[nH]n3)=O)CCCC1N(C(=O)C(c1cncc(F)c1)C)CC2 CC(C)(CCNC(C1CC1(F)Cl)=O)NC(=O)Cc1n[nH]cc1Br CCC(CC(F)(F)F)C(=O)NCC1CCN1C(c1cc2c(C)cccn2c1)=O C(=O)(C(CCC)N(C(=O)CCCCSC)C)NC(CC)CC c1(N2CC(c3scc(C)n3)OCC2)nc2c(c(=NCC3CCCN3C)[nH]1)CCCC2 c1(C(N(CC(C(C)C)C)C)=O)ccc2c(n1)CN(C(c1cn(C)cn1)=O)CC2 C(CC(C)C(=O)NCC1(O)CN(C(c2sccc2CN(C)C)=O)C1)OC c1(C(N2C(C)CCN(C(C3CC4(CC4)C3)=O)CC2)=O)cn2cccc(Br)c2n1 c1(C(N(C(CNC(C2CCC(=O)N2)=O)C2CC2)C)=O)ccsc1Cl N1(C(c2ncsc2Br)=O)CC2C(C1)N2C(c1cnc(C(F)(F)F)nc1)=O C(CC(CO)C(C)C)NC(c1ccc(CNC(C=C(COCC)C)=O)o1)=O C12(C(=O)OC)CC(CNCCC(N3CCCC3C)=O)(C1)C2(F)F CC1(NC(c2nncn2C2CC2)=O)CCCN(C(=O)C(C2CCCCC2)F)C1 c1(OCCC)cc(NCCN(C2CC2)CC2CC2)ccc1OC.C12CCC(C1)OC2.NC CCC(CC)C(=O)NCCCC(C)(C)NC(C1C2CC(=O)CC12)=O C(CCC(O)C(=O)N1CC(CC(C)C)C1)NC(CC1CC(CC)C1)=O c1(C(N(C)CC2CCCN(C(=O)Cc3cnn(CO)c3)C2)=O)nccc(Cl)c1O c1(OCC(=O)N(C(C)CNC(=O)Cc2cncc(C)c2)CC)c(Cl)cccc1Cl N1(C(c2cc(C)oc2)=O)CCCC(NC(c2ccc(Cl)c(C)c2)=O)C(F)C1 C(=O)(C(C)(O)CC(F)F)NCC1CCN(C(Cc2c(C(C)C)cccc2)=O)C1 c1(OCC)ccccc1C(=O)NC1CCC(NC(c2onc(CC)c2C)=O)C1 c1(C(N(CCCCNC(CCC#CC)=O)C)=O)cc(S(=O)(=O)C(C)C)ccc1F c1(CN2CCC3CC(C(N4CC(O)C(O)C4)=O)C3C2)cc2cc(Cl)ccc2[nH]1 c1(C(C(C)NC(=O)CCn2cc(C(c3ccccc3)O)nn2)C)ccc(Cl)cc1 N1(C(C2CC(C)SCC2)=O)CCCN(C(c2cc(C3CCCCC3)on2)=O)CC1 c1(C(N2CCCC(C)(NC(c3n(C)ccn3)=O)C2)=O)cc(F)c2[nH]nnc2c1 O=C1CCC(NCc2ccnn2CCSc2ccccc2)c2ncccc2N1 c1(CNC(C2C(C)C2)=O)cnc2c[nH]nc2c1.CNCCO.C(=O)(NCCOCCO)N c1(C(N(CC(CC)NC(C2CCC2(C)C)=O)C)=O)cnc(O)cc1C c1(CN2CC3C(C(=O)Nc4cn[nH]c4)C3C2)cccc(F)c1Br Cc1cc(F)c(C(=O)NC2(C)CC(NC(=O)C(C3CCC(=O)N3)C)C2)cc1F N1(C(c2scc(OC)c2)=O)CCC(=CCNC(=O)CCC2CC3CCC2C3)CC1 CCC(C)(C)OCC(=O)NCC1CC1NC(=O)CC1(C(=O)C(O)c2cnc[nH]2)CC1 C1(C(=O)N(CCCNC(c2nc(O)sc2C)=O)C)(OCC)CCSCC1 CC(C)C(C)C(C)CC(=O)N1CCC(CN(C)C(c2cc(F)c(Cl)cc2F)=O)C1 c1(C(N2C(COC(C)=O)CCCC2)C(=O)NC2CC2)ncc(Br)cc1F CC(C)CC(=O)NCC(=O)NC1COC(CNC(C2(C(=O)N(C)C)CC2)=O)C1 C1(C(N(C)Cc2nc(C)[nH]n2)=O)CC(C)(C)CCN1C(C1CNC(=O)O1)=O CC1=CC(C(=O)NC(C)CCNC(C2CC2C(F)(F)F)=O)SC1 c1(NC(C2CC(OC)CN2c2cc(N(C)C)ncn2)=O)ccc(O)cc1C N1(C(C2(CSC)CC2)=O)CC(NC(=O)C(C)S)C(C)C1 C1(NC(c2ccc(CC)cc2)=O)CCC2(C1)CN(C(c1c(C)ncnc1C)=O)C2 Cc1oc(-c2ccccc2)c(CN(CC(=O)O)C(C2C3CCCCC23)=O)c1C C1(CC(=O)NCC(C)(C)OCCNC(C2N(CC)CC2)=O)COCCO1 c1(C(N2CCC(C)C2CNC(=O)C2=CCCC2)=O)ncc([N+](=O)[O-])n1C N1(C(CCC=C)=O)CC(C)(C)CC1C(=O)NCC1CC1(Cl)Cl Cc1ccc(C(=O)NC(c2cnn(C)c2)C(=O)NCc2noc(C3CC3)n2)o1 C#CCC(O)C(=O)NC1(C(N2CCC(C)(CO)C2)=O)CCOCC1 CC(C)(C)C(C)(O)C(=O)NC1CC(F)(CNC(=O)CS(=O)(=O)C2CC2)C1 N1(C(C(SC)SC)=O)CC2CC2C1C(=O)NC1COCCOC1 C(C(=O)N(C1(C(=O)NCC2CC(O)C(O)C2)CC1)C)(C(C)(C)C)OC C12(CNC(CC(=O)OC)=O)CC(NC(C3CC(N(C)C)C3)=O)(C1)C(C)O2 C=C=CCCC(=O)N1CC(=C(F)CNC(c2ccccc2SCC(N)=O)=O)C1.SC C1(C(=O)NCC(C(CC)CC)C)CN(C(C2CC(F)(F)C2)=O)C2(CCC2)C1 N1(C(c2c(CC)cno2)=O)CC(CNC(=O)Cc2cccnc2O)C(C)C1 c1(C(C)Oc2cccc(CO)c2)nc2ccccc2s1.C1(C)(C(=O)O)CCCCO1 C(N=c1[nH]c(N2CC3CCC2C3)nc2ccsc12)c1snc(C)n1 c1(C(=O)OC)cc(=NC(C)C(N2CCCC2c2cccc(O)n2)=O)[nH]c(Cl)n1 C#Cc1ccc(C(=O)NC2(CO)CCN(C(=O)C(c3nc(C)cs3)C)C2)nc1 C1(F)(C(=O)Nc2cccc(C3CC3)c2)CCCN(C(=O)C2CC2)C1 N1(C(C(N2CCNC2=O)C)=O)CCCCC(NC(=O)CN2CSCC2=O)C1 CC1CC(CCNC(=O)CCC2CCCOC2)CCN1C(=O)CCn1cccn1 c1(C(N2CCCC(O)(CC3CC3)C2)C(=O)NCC=C)cc(OC)nc(Cl)c1 c1(C(=O)NC(CC)CNC(=O)C(N)=O)cncc(Br)c1Cl N1(C(CC2(CSC)CC2)=O)CCCCCC(NC(C2C(CO)C2(C)C)=O)C1 C12(C(N3CC(N(C(=O)C=CC(=O)NC4CC4)C)C3)=O)CCCC1CCC2 N1(c2cc(N3CCC(OC)C3)ncn2)CC(C)OCC(C)(C)C1 C(=O)(C(C)CC(C)(C)C)NCC1(C(=O)NCC(C)CC2CCCC2)CC(=C)C1 CCCC(C(=O)NCC(C)NC(C1Cc2ccccc2C1)=O)S(N)(=O)=O C1(C)(CNC(CCc2n(C)ccn2)=O)CC(F)(F)CN1C(C1CCCC1O)=O C1(NC(CS(=O)(=O)N(C)C)=O)CCC2(CCN(C(c3ccccc3F)=O)CC2)C1 CC1(NCC2(NC(COC(C3CCC(C(C)(C)C)CC3)=O)=O)CC2)CCOCC1 Cc1cc(C(=O)NC2CN(C(C3CC34CCC4)=O)CC23CC3)cc(C)c1Br Cc1ncccc1C(c1nnnn1C1CC(F)(F)C1)NC1COC1 CC(C)(C)C(CNC(c1ccc(CC2CC2)cc1)=O)C(=O)N1CC2(CC=CC2)C1 C12(C(=O)NC(c3ccn(C)n3)C)CC(CO)(CN1C(=O)CC1CCC3CC13)C2 C(CC(C)(c1nnnn1C1CCOCC1)NCC1CCCOC1)N(C)C C1(NC(=O)NCCN(CCNCC)C)CCCCC1 c1(NC(CC(N)c2cncs2)=O)ccc2cc(Br)ccc2c1 C(=O)(C1=CC2C=CC(C1)C2)NCC1OCC(CNC(c2c(C#C)cn(C)n2)=O)C1 C(CC(=O)N(C)Cc1nnc(C)o1)(C(C)CC)NC(C=CC(CC)C)=O c1(C(=O)NCCCN(C(C2CC(C)C2(C)C)=O)CC)ccc(N)c2ccncc12 c1(CC(=O)NC2CC3(C(NC(C4N(CCC)CCC4)=O)C3)C2)cc(F)cc(Cl)c1 C1(O)(C(=O)NCC2C(C)CN(C(C3CCC(C(N)=O)O3)=O)C2)CCN(C)CC1 C1=CCCC(CSCCOCC(c2nnnn2CCCF)C2CC2)CC1 C(=O)(C(C(C)C)OC(C)=O)C(c1cc(OCC)no1)=O.N1(C(C)=O)CC(O)(CN)C1 C#CCC(C)(C(=O)NCC(O)CN(C)C1CC1)NC(C1CCCC12CC2)=O C1(O)(CNC(CSCC#C)=O)CCCN(C(c2ncn(C)c2C)=O)CC1 C1(C(=O)NC2CC(NC(c3ccsc3C(F)F)=O)C2)Cc2ccccc2CO1 C=C(C)C1CN(C(=O)CC2CN(C(c3c[nH]cc3C)=O)CCC2C)CCO1 c1(C(=O)OC)nc2c(s1)N(C(C1CCCCC1n1cccc1)=O)CCCC2 c1(C(N2CC(N(C(=O)Cc3ccon3)C)C(F)C2)=O)cc2ccccn2c1 CC1CN(C(c2cccc(F)c2F)=O)CCN1C(=O)CN(C)C C1(CN(C(=O)C(C2(O)CCC2)NC(=O)C=Cc2nccs2)C)CCCOC1 N1(C(C2(OC)CC2)=O)CC(C)(CCC(N2CCC(OC(F)F)C2)=O)C1 C#CCCCCC(=O)NCc1nc(C)c(C(N2CC3C(C)C3C2)=O)o1 N1(C(Cc2cc(C)n(C)n2)=O)CC2CC(C(=O)NCCN(C)CCO)(C2)C1 c1(C(=O)NC2CCCCN(C(C3C(C#N)C3)=O)C2)nnn2c1CSCC2 N1(C(C(CC)OCC)=O)CCN(C(c2ccnc(C3CC3)c2)=O)CC1C(C)(C)C c1(CN(C(C2CN(C(=O)OC(C)(C)C)C2)=O)CC)cn(C)nc1-c1nn[nH]n1 N1(C(C(C(C)C)OC)=O)CCCCC(NC(C2CCC(N=[N+]=[N-])C2)=O)C1 C1(C(=O)NC(C2CN(C(c3ccncc3Cl)=O)C2)C)CCCC1(C)C c1(C(=O)NC2(CNC(c3c(C)ocn3)=O)CCC2)cccc(C2CC2)c1 C1(C#N)(C(N2CCC(CN(C(C(C)C3CC3)=O)C)CC2)=O)CC2CC2C1 N#CC1(C(=O)NC2COCC2C(N2CCC(OCC(N)=O)C2)=O)CC12CCC2 C(c1ccc(-n2ccnc2)cc1)=CC(=O)N(C(C)C)CCN(C)C(C1CC1Cl)=O C1(C(=O)NC2CC(NC(C3(NC(=O)C(F)(F)F)CC3)=O)C2)CC1C1CCCC1 N1(C(C2C(C(C)C)CCO2)=O)Cc2[nH]nc(C(N3CCC4(CCCC4)C3)=O)c2C1 N1(C(CCC2CCCN(C(C3CCC(N(C)C)C3)=O)C2)=O)CCCOC(C)(C)C1 C1(CCC(=O)N(C(C(=O)N(CCOC)CC)C)CC)CCC(=O)C1 c1(C(C)=O)cccc(OC(C)C(=O)NC(C)CNC(c2conc2C)=O)c1 C(C1CCCCC1)=C(C(N1C(CN(C(CC2(OC)CC2)=O)C2CC2)CCC1)=O)F C1(C)(C(=O)NC(C2(C)CC(NC(C3C4CCCC34)=O)C2)=O)CC2CCC1C2 N1(c2cc(C)nc(CC3CC3)n2)CC2(C)CN(C(c3cc(C)sn3)=O)CC2(C)C1 CS(=O)c1ccccc1CC(=O)NCC1C=CC(NC(c2csc(CO)n2)=O)C1 c1(NC2(CC(=O)OC)CC2)c([N+](=O)[O-])ccc(Cl)c1C CC1CN(C(C2CC2c2cccnc2)=O)CCCN1C(c1cc(CF)on1)=O N(C1c2ccccc2CC1NC(C1(C)CCCC1)=O)C(CCC(C)OC)=O C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(C2CCN(C)CC2)=O)CC12CCC2 c1(OC(C)=O)cccc(C(N2CC(NC(=O)C(C)(C)n3cccn3)C(F)C2)=O)c1 N1(C(C23C(C)OC(C)(C2)C3)=O)CC(NC(c2cncc(O)c2Cl)=O)C2(CCC2)C1 N1(C(CSCCCC)=O)CCCC1CCCNC(c1cnc(C(C)C)o1)=O C12(Cc3n(CC(=O)N(C4CC4)CC)c(S)nn3)CCC(N)(CC1)CC2 C1(CC(=O)OC)CN(C(=O)Nc2cnc(Sc3ccccc3)[nH]2)CC(CC)O1 c1(CCOC)ccc(S(=O)(=O)NC2CC2(c2cccc(C)c2)C)s1 N1(C(CCCC2C(C)C2)=O)CCCC(N(C(=O)C=Cc2cc[nH]c2)CC2CC2)C1 c1(C(N2CCN(C(=O)Cc3ccon3)C3C2C3)=O)ccc2c(c1)CCC2 CCCC(CC)NC(c1cn(CC2CCCO2)nn1)c1nnnn1C(C)(C)C C1(CC#C)(C(=O)NC2(CCNC(=O)CC(O)C3CCCC3)CC2)CCCO1 c1(Cn2cc(C3CCN(C(c4n[nH]cc4I)=O)C3)nn2)c(F)cccc1F N1(C(C(C)CCN(C)C)=O)CCN(C(=O)COc2cccnc2Cl)CC(O)C1 c1(C(C)C)ncncc1C(=O)N(CC(C)NC(C1CN(C)C1)=O)C c1(OC)cc(F)ccc1SCC(c1ccccc1)=O.C12CC(CN1SC)OC2=O c1(CC(=O)NC2CCN(C(C3C(CCC)CCC3)=O)C2)cc(C)cc(F)c1 C(C(=O)NCCCC1CC1)(C1CCOC1)NC(=O)CSC(F)F c1(NC(=O)NCCc2cn(CC)nc2)cccc(OC)c1Cl C(=O)(C1CCCc2sccc21)NC1CN(C(CS(=O)(=O)N(C)C)=O)CC2(C1)CC2 N1(C(c2nc(C#C)sc2)=O)CC(NC(=O)CC(=O)OC)CC12CCCCC2 N1(C(CC2(C)CCOC2)=O)CCN(Cc2ccc(F)cc2)CC1.N12CCCC1C2 N1(CC2(C#N)CCC2)CC(=O)N(Cc2cnn(-c3ccccc3)n2)C1=O C#CCCC(=O)NCCC1CCC(NC(c2ccnn2C(C)C)=O)C1 C(CNC(c1cnncc1Nc1ccn(CCF)n1)=O)(CC(=O)NC(C)C)OC N1(C(c2cc(OC)cc(Br)c2)=O)CCN(C(=O)NCc2csc(C)n2)CCC1C N1(C(CCC#N)=O)CC2CCC1CN2C(c1cc(C(F)(F)F)cs1)=O c1(OCC(N2CC(CNC(C(C#C)(C)C)=O)C2)=O)c(C)cccc1Cl C(C(C)CN=c1ccc(S(C)(=O)=O)c[nH]1)NC(c1c(C(C)C)nns1)=O N1(C(C(=O)Nc2c(C)scc2)=O)CC(N)CC(O)C1 Cc1nsc(Br)c1C(=O)NC1CCCCC1NC(C1CCSC1)=O c1(C(=O)NC(C2CCCC2)CNC(C(CC#C)C2CC2)=O)cccn2nncc12 c1(C(N(CC(CC)NC(C=C(CCC)C)=O)C)=O)cc(C)cc(O)n1 N12CCC3(CC3C1)C(=O)NCC2=O.C(=O)(CCCc1nc(C(F)F)no1)NC1CC1 c1(OCCN(C2CCC(=O)NC2)C)cc(Cl)cc(Cl)c1.C12CCN(C1)C(=O)C(=O)N2 n1(C[Si](C)(C)C)cnc(=NC(=O)C(=O)NCCCOc2cc(F)cc(Cl)c2)[nH]1 C1(O)(CNC(C(C)=C2CCC2)=O)CN(C(c2cnc(C(C)(C)C)o2)=O)C1 C(CCN=c1[nH]c(N2CCCN(C(N)=O)CC2)nc2cc[nH]c12)OC(C)(C)C N1(C(c2cc(C)nc(O)n2)=O)CCOC2(CCC(NC(=O)C#CC3CC3)CC2)C1 C1(C(=O)NCCS(CC)(=O)=O)CCCCN(C(C2CC(=O)NC(=O)C2)=O)C1 c12cc(N)c(s1)c(=O)[nH]c2=O.c1(COC)c[nH]c(C(=O)O)c1 C1(NC(CC2CCN(C(C(C)n3cccn3)=O)C2)=O)CC(F)(F)C1(C)C C(CNC(=O)CC1CC=CC1)(CC(=O)NCC1(C)CC(C)=NO1)OC c1(C(=O)NCC(C2CCC2)NC(COC)=O)cc(C2CCCCC2)ccn1 C1(C(NOCC2(C)CC2)=O)CCCCN1C(c1coc(C(F)F)c1)=O N1(C(C(C)S(N)(=O)=O)=O)CC(NC(c2cnc(O)nc2O)=O)CC(C)(C)C1 c1(C(=O)NC(C2(O)CN(C(c3cc(OC)no3)=O)C2)C)cc2ccccn2c1 N1(C(C(C)OC2CCCC2)=O)CCOCCC1C(=O)N(CC(F)Cl)C c1(C(=O)NCC(CC)NC(CC(=C)I)=O)ccn(C)c(=O)c1 C1(C#N)(C(=O)NCc2scc(CNC(CCCN(C)C)=O)n2)CCCOC1 C1(NC(C2(C)CC2(F)F)=O)CN(C(=O)CNc2nccs2)Cc2ccnn2C1 Cc1nn(CC(N2CC=CC2CNC(=O)COc2cccc(F)c2)=O)cc1Cl N1(C(=O)Nc2cccnc2)CCC(O)(CNc2cc(CO)cc(Cl)c2)CC1 C=CCC(F)(F)C(=O)N(C(=O)CCc1cccc(O)c1)C1CC1C(=O)OC C(=O)(C(C)(F)C(=O)N1CC(NC(=O)C=C(C)CN2CCOCC2)C(C)C1)OCC C1(CC(=O)OC)CCC1NC(=O)CCC1CC(NC(=O)OC(C)(C)C)C1 C1(OC)CC(NC(c2ccncc2O)=O)C12CCN(C(=O)C=CCF)CC2 CCCCCCC(F)C(=O)NC1(CO)CCN(C(=O)C2=CCCCC2)C1 C(=O)(C(C)(O)CCN(C)C)NCC(C)CNC(=O)C(F)=C1CCCC1 c1(OC(c2cccc(C34CCC(NCC)(CC3)C4)c2)=O)ccc([N+](=O)[O-])cc1 C=CCCCC(C1CC1)NC(=O)CC1CCCN(C(C2CCCC2F)=O)C1 c1(NC(=O)NC(c2ccc(F)cc2)C(F)(F)F)cnc(Cl)cc1Cl Cc1ccnn1CC(N1CCCC1CNC(C1C2CCCC12)=O)=O C(=O)(C(C)C(C)C(C)(C)C)N1CC(CCCCNC(C=CCN(CC)CC)=O)C1 c1(C(N(CCC(=O)NCC(=O)NCC)C)=O)cc(CO)n[nH]1 c1(C(=O)NC2(C)CCCN(C(=O)CCc3cnoc3)C2)cnc2cccnc2c1 Cc1cccc(Br)c1C(=O)NCC1(C)CCN(C(c2c(C)cnn2C)=O)C1 c1(C(=O)NCCCOCCNC(CC(C(C)C)C)=O)cnn2c1OCCC2 C1(C(=O)OC)NC(=O)C2CCC1N2C(=O)C(N1CCSCCC1C)=O c1(CC)noc(C)c1C(=O)NCC(C)C(=O)N(C)CCN1CCOCC1 N1(C(Cn2c(C)ncc2)=O)CC2CCCC2(C(=O)NCCN2CCCOCC2)C1 c1(C(=O)NC(CC(C)NC(c2cn(CC)nn2)=O)C)coc2c1CCCC2 c1(C2C(C(=O)NCC(CCOC)NC(=O)C(C)O)C2)ccncc1F C1(C(=O)NCC2CC(NC(c3c[nH]c(=N)s3)=O)C2)CC(=O)c2cc(Cl)ccc2O1 C1(NC(c2ccc(CC)[nH]2)=O)CCOC(CNC(c2cc(OC)c(Cl)s2)=O)C1 C1(N(C2CCC2)C(C2CN(C)C(=O)C2)=O)CN(C(C2CC(C)(O)C2)=O)CC1(C)C CONC(=O)C(=O)N1CCC(C(=O)NCCCSC(F)F)C1C(C)C N1(C(Cc2n(C)ccc2)=O)CCC(CCCNC(C2CCC23CCC3)=O)CC1 C(CC(C)(C)C)(C(=O)N1CCC(NC(=O)CCc2ccccn2)C1C(C)C)OC CC1CN(C(c2ccsc2Cl)=O)CCC1NC(=O)CNC(=O)C(C)(C)C c1(C(N2CCC(N(C(C(C3CCOCC3)OC)=O)C)CC2)=O)ccc(Cl)cc1F CON1CCC(N(C)C(C2CC(NC(=O)CC3CCC(O)C3)C2(C)C)=O)CC1 C1(CNC(C2C(C)(C)C2(C)C)=O)C(C2CC2)CCN1C(C12CC(CO1)C2)=O C(CC(C)C(=O)NC1(C2CCCN2C(=O)C(=C2CCCCC2)F)CC1)OC c1(C(=O)NCCCCCN(C)C(C2CSCCS2)=O)ccn2cncc2c1 C(=O)(C1=Cc2ccccc2C1)N1CCC2CN(C(C=CC(CC)C)=O)CC2C1 c1(C(=O)NC2CN(C(C3CC(SC)C3)=O)CC2N=[N+]=[N-])cnc2[nH]nc(O)c2c1 C1(CNC(C2N(C(C)=O)CCCC2)=O)(NC(C2CC(F)C2)=O)CC2CCC1CC2 N1(C(=O)OC(C)(C)C)CCC(c2ccccc2)(NC(c2nn[nH]n2)=O)CC1 C1(C)(NC(c2c(C)cn(C)c2)=O)CCN(C(=O)Cc2c(C)n[nH]c2C)CC1 N1(C(C2CC(C)(O)C2)=O)CCN(C(=O)CC2(C#N)CCOCC2)CC(O)C1 N1(C(C)C(=O)NCC(O)CN(C)C)CCCC(C)(NC(c2ccccc2F)=O)C1 C1(NC(c2c(CC)n[nH]c2)=O)CC2(CCC(NC(c3c[nH]ccc3=N)=O)CC2)C1 C1(NC(C(C)CC23CC(C2)C3)=O)C2CCCCCC12.C(C)(C)(C)OC(=O)O C1(NC(=O)CCCOc2cccnc2)C2CCN(C(C3(F)CC3)=O)C12 C(C(C)(C(=O)N1CCC(O)(CN(C)C(C23CC4CC2C3C4)=O)C1)OC)OC N(C1CCCc2cc(Cc3ccccc3C#N)ccc21)C(N(C(C)C)C)=O N1(C(C2C(C)(C)CO2)=O)C2CCC(C2)C1CNC(=O)C=CCO N1(C(C=CCCC)=O)CCC=C(C(=O)NCCCCCSC)C1 CC(C)(CC(F)F)C(=O)N1CCCC(CNC(C2CCC(=O)C2)=O)C1 C(=O)(CC1=CCN(C(=O)C(C)C)CC1)NCc1c(C)nc(F)cc1 CCCC(O)C(=O)NCC1CC(NC(C2CC(F)C2)=O)C1 c1(CNC(C(C)c2ccsc2)=O)ncoc1C1CN(C(c2ccccc2)=O)C1 N1(C(C(CSC)(C)C)=O)CC(CNC(=O)CCc2ncccc2C)C2(CCC2)C1 N1(C(CC2CC(=O)C2)=O)CCCCCC1CNC(c1cccc(OCCF)n1)=O c1(CCNC(C(C)N(S(CCCC)(=O)=O)CC)=O)nnc2n1CCC2 N1(C(CNC(=O)OC(C)(C)C)=O)CCC(C)(CNC(c2ccc(C(F)F)o2)=O)C1 C1(CNC(C2(CC)CC2)=O)CN(C(C2CCOC2C)=O)CC1C(F)F Cc1c(C(=O)NC2CC(O)CN(C(=O)C(C)(C)C(F)F)C2)sc2ccccc12 C1(CNC(C2(O)CC(C)(C)C2)=O)CN(C(=O)Cc2cccc(Cl)c2)CC12CCC2 c1(C(=O)NCCNC(CN(CCCOC(CC)C)CC)=O)ccc(F)cc1F N1(C(CCN(C)CC)=O)CC(N)C(NC(C2(COC)CC(F)(F)C2)=O)C1 C1(C(=O)NC(CC)COC)CC2CCC(C1)N2C(c1ccc(C)nc1C)=O N1(C2CCN(CC=C)C2=O)CCC(NC(=O)C(CC)OC)C(CO)CC1 N1(C(CC(C)C)=O)CCC(NC(=O)C(C(C)C)n2cccc2)C2(CCC2)C1 c1(CCNC(C2(N(C(C3C(C(=O)OC)C3)=O)C)CC2)=O)ccnc(O)c1 N1(C(c2c(C(C)C)cco2)=O)CC2CC(NC(C3CN(S(C)(=O)=O)C3)=O)CC1C2 c1(C(=O)NCC2N(C(CC=CC)=O)CCOC2)ccc(OC)nc1OC C1(N(C)C)CCC(N=c2cccc(S(=O)(=O)NCC3OCCOC3(C)C)[nH]2)CC1 CC1(C)COCC(C)(CNC(=O)C(N)CCF)C1 c1(CC)ccc(Cl)cc1NC(C1CN(C(c2cnc(O)c(F)c2)=O)CC1C)=O C1(C(N2C(C)(C(=O)OC)CC2)=O)CC(C)(C)CN1C(c1cc(F)n(C)n1)=O c1(CN2C(c3ncc(-c4ccc(C#N)nc4)[nH]3)CCC2)cc(Br)cc([N+](=O)[O-])c1 C1(C(N(CCCNC(C2(C#N)CCOCC2)=O)C)=O)CCc2ncccc2C1 C1(CCNC(c2c(C)[nH]cc2)=O)CN(C(=O)Cn2ncccc2=O)CCCO1 c1(C(=O)NCC2(NC(C3CC3F)=O)CC2)cc(Cc2ccc(Cl)cc2)ccc1O C12(NC(CCC=CC)=O)CC(C1)N(C(c1[nH]c(O)nc1C)=O)C2 c1(C(N2CCC(O)(CCNC(c3c(C)coc3)=O)C2)=O)coc(S(N)(=O)=O)c1 c1(CCC(=O)NC(C2CN(C(=O)CC(=O)N(C)C)CCO2)C)nnc(S)n1C C(=O)(C1=Cc2ccccc2C1C)NC1(CCCNC(C(C(C)C)C)=O)CC1 C(=O)(C(O)CC(C)(C)C)NC1C(C)N(C(=O)CC(C)(C)C)C(C)C1.n12cc(nn1)C2 CCC(C)(C)CCCC(=O)NC1CC1NC(=O)Cc1ccnc(Cl)c1F N1(C(Cc2nnc(C)o2)=O)CCC2CCN(C(C3(C#N)CCCOC3)=O)CC12 c1(OC)ccc2[nH]cc(C(=O)NC3CC(C)N(C(C4CCCC4(F)F)=O)C3)c2c1 N1(C(C2(O)CCC(CC)C2)=O)CC2CC(C1)CN(C(=O)CCCC(N)=O)C2 c1(C(N(CCCN(C(C2(C)C(C(=O)OCC)C2)=O)C)C)=O)occ2c1CCOC2 CCC(C)CC(=O)NCCCC1CCCN1C(=O)CCCCc1ccc(F)cc1 C(CN=c1nc(Cl)[nH]c(C)c1C#N)=CCNC(C(C)OCCCC)=O N1(C(Cc2cncc(C)c2)=O)CCC(NC(=O)C=CBr)C(O)C1 C(=O)(C1=COCCO1)NCc1cn(C2CCN(C(CC(CC)C)=O)C2)nn1 C1(C)(COCC)CCN(C(C2(c3nnnn3C3COC3)CC23CCOC3)=O)CC1 N#CC1=C(C(=O)NC2CCCC2CC(N2CC(N3CCOC3=O)C2)=O)CCC1 C1(C(N(CCN(C(C)C)C(c2scnc2Cl)=O)C)=O)CCCC1CF C1(NC(C=C(CC)CC)=O)CCC2CC1CN2C(c1ncn(C)n1)=O C1(C(=O)NCC2CCC3CN(C(=O)C4=CCSC4)CC23)CC2CCCCCC12 N1(C(C)=O)CC2CCC1C(NC(=O)C(C)CSc1ccc(C)cc1)C2 CCCCC(C)(F)C(=O)NCC1CCC(CNC(=O)C(C)(C(C)C)OC)CC1 c1(NC(C2CCN(C(c3cc(OCC)n[nH]3)=O)C2)=O)ccc(CN(C)C)cn1 C=CCC(C)(C)CNC(C1(NC(=O)CC2CCC(=O)NC2)CCSC1)=O C1(C(=O)NCCN(C)C)(NC(C=C(COC)C)=O)CCCC1C C1(C(=O)Nc2cn(C3CC3)cn2)CCN(C(C2CC(F)C2)=O)CC1O C#Cc1ccc(C(=O)NCC2CCN(C(C3(C)CC3)=O)CC2C)c(Cl)c1 N(C1CS(=O)(=O)Cc2ccccc21)C(=O)NCC(C1CCOCC1)C N(C1c2ccccc2CC1NC(=O)CC1CC2CC2C1)C(C(F)=CC)=O N1(C(C(C2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C)=O)CC2CCC(C1)C2O C1(C)(CNC(c2c(C)scn2)=O)CN(C(C2CC(=O)OC2(C)C)=O)CCO1 C1(NC(C)=O)CCC(C(N2CC(C(C)NC(=O)CCc3nc(O)n[nH]3)C2)=O)CC1 c12ccc(cc1)CC(=O)NC2.c1(C(C)C)cc(C(=O)OCC2CCCO2)no1 Cc1nc(C(=O)NC(C2CCCN(C(C3CC(N(C)C)C3)=O)C2)C)sc1C C1(NC(c2c(CC)occ2)=O)CCN(C(c2c(Cl)cnn2CC)=O)C12CCCC2 C(=O)(C(F)(CNC(=O)C(F)(F)C=C)C(C)C)NC(C=C)(C)CC N1(C(c2c(C)onc2)=O)CC2CN(C(=O)C(C)Sc3ccc(Cl)cc3)CC2(C)C1 CN1CCC2(CCC2)C(Nc2cc(F)c(OCCC(=O)O)c(F)c2)C1 C(CCCC(=O)NC)NC(c1n(CC=C)nnn1)c1cnn(CCC)c1 Cc1ccc(N)cc1C(N1CCN(C(=O)C(c2ccccc2)F)C(CCO)C1)=O C(C1=NOC2COCC12)NC(C(CC(=C)C)NC(=O)Cc1ccnn1C)=O c1(C(N2CC(CNC(C(C)CCN(C)C)=O)C(F)(F)C2)=O)cc2cccn2cn1 Cc1nc(=N)[nH]c(=NC(C)CN(C(=O)C=CCN(C)C)C)[nH]1 c1(NC2CCN(C(c3c(OC)cnc(F)c3)=O)CC2C)cc(O)nc(=O)n1C N1(C(C(c2ccccc2)OC(C)=O)=O)CC2CC1CC2N1CC(C)(OCC)C1 C1(N(C(=O)CCC2(C#N)CCC2)CC)CCCN(C(=O)C(C)c2ccsn2)CC1 N1(C(COC(CC)C)=O)CCCC(N(C(=O)CCC2C(=O)ON=C2C)C)CC1 N1(C(C2C(C)(C(C)C)C2)=O)CC2CCC1C1CN(C(=O)CCOC(=O)N(C)C)CC21 C12(CNC(c3cc(SC)oc3C)=O)CCCCC1N(C(=O)C1=COCCC1)CC2 c1(C(=O)NC(C)C(=O)NC2CCNC2=O)ccc2c(c1)CC2 CC1CCc2c(C(=O)NCC(CNC(=O)CN3CC(C)(C)C3)CO)csc2C1 C1(C)(C(N(CCCNC(c2cc(C)ncn2)=O)CC)=O)CCNC(=O)C1 C1(CNC(C(C)=CC)=O)CN(C(=O)Cc2ccco2)C2CC12 c1(OCCC(C(=O)N2CC(OCC)(CO)C2)OCC(=O)OC)ccc(F)cc1 c1(C(N(CCCN(C(CC(=O)NCC#C)=O)C)C)=O)c[nH]c(=O)c2ccnn12 c1(C(=O)NC2C(NCc3scc(C(=O)OCC)c3)CCC2)ccc(F)c(F)c1 c1(C(N(CC(C)NC(=O)CC(C)(O)C2CC2)C)=O)cccn2nnnc12 c1(C(=O)NC(CC=C)CNC(c2sc(Br)cc2F)=O)nn(C)c2c1CCC2 O(N=C1CCCCCC1)CC(N1CCC(N(C(C(C)=C(CC)C)=O)C)C1)=O CC1CCN(C(c2ccsc2)=O)C(CNC(C2CCN(C(=O)OC)CC2)=O)C1 c1(C(N2CCSCC2)C)cn(CC2CCCOC2)nn1 c1(C(=O)NC(c2cnn[nH]2)C)cccc(CNC(C2(C)CCCC2)=O)c1 C(=O)(C1=CC2(CCN(C(c3ccnn3CC)=O)C2)C1)NCCC(CC)(F)F CC1(C)CCC(C(=O)NCC(CNC(=O)Cc2csc3nccn23)CO)CC1 c1(C(=O)NCC(CC)NC(c2ccc(CO)cn2)=O)cnn2c1OCC2 CCCCCCC(F)C(=O)NCC1CCCN(C(=O)CCNc2cncnc2)C1 C1(NC(C(C=C)O)=O)CC2CCC1C(NC(c1ncnc(C)c1OC)=O)C2 c1(C(N2CCCC23CC3)C(=O)NC2C(C)C2)ccc(C(=O)Nc2nnn(C)n2)cc1 C1(CC=C)(C(=O)NCC(F)CNC(C2(COC)CCCO2)=O)CC=CC1 CC1CN(C(=O)CC2CC(C3CC3)C2)CCN(C(c2cc(O)cc(=O)o2)=O)C1 C1(CNC(c2cc(Cl)c[nH]2)=O)CC2(CCN(C(C3CCCCC3(F)F)=O)C2)CO1 c1(NC(C(C)=C(C)C)=O)ncccc1C(=O)NCC1(c2ccon2)CC1 C(=O)(C(Cc1ccccc1)S(C)(=O)=O)NCCNC(C(c1cncc(F)c1)C)=O c1(CC)ccc(C(=O)N=S(C)(=O)c2ccccc2Cl)c2c(=O)c(CC)c[nH]c12 Cc1ccc(CNc2cnc(Cl)cc2C(N2CCCC2CO)=O)c(Cl)c1 N1(C(C(C(C)(C)C)c2nn[nH]n2)=O)CC2(CCC(=O)NC2)C1.C1CCC1 c1(CNC(Cc2snc(CC)n2)=O)nccc(Cl)c1F c1(N2CCC(CNC(c3c(C)cccn3)=O)C2)nnccc1C#N C(C)(CCC(=O)N1CCC(NC(C23CC(C(C)(F)F)(C2)C3)=O)C1)OC NC1CC(C(N2CCC(c3cc(O)no3)CC2)=O)C12CCOCC2 N1(C(c2sc(CC)c(C)c2)=O)CCN(C(C2CCCCS2)=O)CC2(CC2)C1 c1(OC)cnc(NC2CCCCC2NC(c2cc(C)ccc2Cl)=O)nc1C C#CC1CCCC1NC(=O)C=CC1CCCN1C(=O)CCCN(C)C C(=O)(CCCC(=O)N(C)C)NCCC(C)N(C(c1c(C(C)=O)cn(C)n1)=O)C C1(CN(C)Cc2nn(C)cc2Cl)CCN(C(=O)CCNC(=O)C(C)(C)C)CC1 C1(NC(c2ccc(OCCC)nc2)=O)CN(CCOCCOC)CCC1C CCC(C)C(CN(C)C)C(=O)N1CCCC1c1ncccn1 c1(NC2(CNC(=O)C=Cc3ncc[nH]3)CCC2)cc(C(N)=O)nc(Cl)n1 N1(C(C2C(OC)(OC)CC2)=O)CCC(C(=O)NC(C)C(=O)OC)C12CCC2 N1(C(CN2CC(C)C2)=O)CC2CC2(NC(c2csc(CS(C)(=O)=O)n2)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)NC(C)CCNC(=O)CCC1CCCCC1 N1(C(C2(CCOC)CC2)=O)CCC(O)(CN(C(=O)C(C)C(C)O)C)CC1 Nc1ccc(C(N2CCCC(NC(c3cccc(CCF)c3)=O)C2)=O)nc1Br c1(C(N2CC3CC(NC(c4cc(Br)n[nH]4)=O)C3C2)=O)cnc2occc2c1 N1(C(c2cc(C)[nH]n2)=O)CCCC2(CCCN2C(C2CC(C)(C)CN2C)=O)C1 N1(C(CSCCC=C)=O)CCCC(N(C(C2CCN(C(=O)NC)CC2)=O)CC)C1 Cc1ccc(NC(=O)C(F)C(C)CNC(=O)CCOCC(F)F)cc1F c1(C(N2CCOCC(NC(C3CC(=O)NC3)=O)C2)=O)nc2ccccn2c1F Cn1ccc(=O)c(C(N2CCC(NC(c3ncncc3F)=O)C(O)C2)=O)c1 N1(C(C2CN(C(C)=O)C2)=O)CCC2(NC(c3cc(-c4ccco4)[nH]n3)=O)CC2C1 c12c[nH]c3ccc(cc13)[nH]c1ccc2cc1C(F)(F)F.N1(CC)CCCCC1CO Cc1nc(O)c(C(N2CC(CCc3cn(-c4ccncc4)nn3)C2)=O)cc1Br c1(CCNC(NCC2(OC)CCOCC2)=NCC2CC2)noc2cc(F)ccc12 c1(C(=O)NCC2(O)CN(C(CC)=O)C2)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 c1(CCC(N2CC(OC)(CNC(c3csc(C(N)=O)n3)=O)C2)=O)nnc(S)n1C CC(c1ccccc1Cl)=CC(=O)N(C)CC1CCCN1C(c1n[nH]cc1F)=O C1(NC(C(C)N(C)C)=O)CC2CC(NC(c3cnnc(O)c3)=O)CC2C1 N1(C(C2(C)CCC2)=O)CCCC(C2CCN(C(=O)C3Cc4ccccc43)CC2)C1 CC(CC(F)(F)F)OCOC(=O)OCC1CCN(Cc2ccccc2)C1 CC(CS(C)(=O)=O)C(=O)NCC(O)CNC(c1cn2ccnc2s1)=O c1(C(N(C(C)CNC(=O)C(C)(C)OC)CC)=O)ccc2c(c1)CCCCN2 C1(C(N2C(C(C)C(=O)NCc3ccccc3Cl)CCC2)=O)CCC(=O)N(C)C1 C1(C(=O)NCCCC(C)NC(C2(C#N)CCCO2)=O)(C(C)C)CNC(=O)C1 CN1N=C(C(=O)NCC2CN(C(=O)CCS(C)(=O)=O)C3COCC3O2)CCC1=O c1(C(N2CC(CNC(C(C)(C)NS(C)(=O)=O)=O)OCC2)=O)cc2c[nH]cnc-2n1 C1(CCOC)(NC(=O)CC(F)(F)F)CCN(C(=O)C(F)Cc2ccccc2)CC1 C(=O)(C(C)(C)CC(=O)NCC1(NC(c2nn(C)c(C)c2Cl)=O)CC1)OC N1(C(C2C3CCCCCC23)C(=O)NCC=C)CCCC2(C1)CN(C)C(=O)O2 C1(NC(C2CC23CC3)=O)CCCC2CN(C(=O)CC(O)C3CC3)CC12 CC12CSCC1CN(C(C1(F)CCN(C(c3cccc(Cl)c3)=O)CC1)=O)C2 C#Cc1ccc(C(N2CCC(NCC3(C)CC3)CC2)C(=O)NCCN(C)C)cc1 C(=O)(CCS(N)(=O)=O)NC1C(NC(C2C(c3n(C)ncc3)C2)=O)CC1 C(=O)(CC1CS(=O)(=O)c2ccccc21)NCCC1N(C(CCC)=O)CCSC1 C12(C(=O)NC(COCC)C)CC(CO)(CN1C(=O)C(O)C(F)(F)F)C2 C1(NC(CCc2cnc(C)nc2O)=O)CC(N=c2ccc3ncc[nH]c-3n2)C1(C)C CCCCC(CNC(c1cc(C)oc1C(F)(F)F)=O)NC(=O)CC(C)CN(C)C CCC(CC(=O)NCC(C1CCCCC1)NC(c1nc(Cl)cs1)=O)c1ccccc1 c1(OCCC)cccc(CC(=O)NC2CC(C)(CNC(=O)CC(C)SC)C2)c1 c1(CC(=O)NCCC(C)N(C(C(CC=C)CC)=O)C)ccc2c(c1)CCO2 C1(C)(C(N2CCCC(C)(NC(C3C4COCC34)=O)C2)=O)CCCNS1(=O)=O N1(C(C(=O)NC(c2ccccc2)C)=O)CSCC1CN1CCC(c2nn[nH]n2)C1 C(=O)(C(C)(F)C(=O)NCCCNCCOCCC(=O)NCCSC(F)F)OC c12ncccc1OC(C)C(=O)N2.C(=O)(C(COC)CC1CCCC1)OC c1(NC(C2C3CN(C(C4CC4c4ccccc4)=O)CC32)=O)cc(Br)c(O)c(Br)c1 c1(OCC(=O)NC)ccc(C(N2CC(Cc3cn[nH]c3)C(C)C2)=O)cc1OC c1(OCC(=O)N(C2CCN(C(=O)Cc3ccsc3Cl)CC2)C)cncc(Cl)n1 C1(C(=O)NC2(CNC(CCc3c(C)noc3Cl)=O)CC2)CCS(=O)(=O)C(C)C1 Cc1nc2n(n1)CC(C(=O)NC(C)CC1CN(C(=O)OC(C)(C)C)C1)CC2 c1(C(=O)NC2(C)CCN(C(c3nc(C)oc3)=O)CC2)cc2nc(Cl)ccc2o1 C1(CNC(C=CC)=O)CCC12CCN(C(=O)CCOCC(F)(F)C(F)F)CC2 N1(C(=O)Cc2cscn2)CCCC(C2CCN(c3ccnc(CO)n3)C2)C1 c1(CN(CCCC(=O)OC)C2CC2)cnc(O)cc1OC C1(NC(C(CC)n2cncn2)=O)CCN(C(c2cc(SC)oc2C)=O)C1C(C)C c1(OCC)ccc(C(=O)NCC2CN(C(=O)C=CCN(C)C)CC2(C)C)cc1C C1(C#N)(C(=O)NC2CC(CCC(=O)NC(C#C)CC3CCCC3)C2)CCOC1 N1(C(CC(=O)OCCC(C)C)=O)CCC(C)(CNC(C2CC(=C3CCC3)C2)=O)C1 C1(CNC(C(C=C)O)=O)CCCCN(C(c2nc(C)[nH]c2C(F)(F)F)=O)C1 C1(NC(CC(CNC(C2C(CC)C2)=O)OC)=O)CC(C)(C)C12CCC2 N1(C(C(C)OC)=O)CC(NC(=O)CN2CCCCS2(=O)=O)CC(F)C1 C1(C(=O)NCCC(=O)NCCC(F)(F)F)(OC)CCCOC1 Cc1cnc(N2CCCC2)nc1C.C12CCC1CN(C)C(=O)NC2=O c1(C(=O)NCC2N(C(C(C(C)C)N3CCCCC3)=O)CC2)cnc(O)n(C)c1=O C=CC(CC)CC(=O)N1CC=CC1(C(=O)NC)COC c1(C(=O)OC2CN(C(=O)OC)C2)ccc2nnc(C(F)F)n2c1 C1(NC(=O)C(c2ccc(Cl)cc2)O)C=CCN(C(C2(F)CC=CC2)=O)C1 N1(N(C2CCCN(S(C)(=O)=O)C2)C(C2C3CCC(=O)C32)=O)CC2(CCC2)C1C1CC1 N1(C(C2N(C(C(CC(C)C)=O)=O)CC(F)(F)C2)=O)CC2(CCC(C)OC2)C1 C1(NC(C2CCCOC2)=O)CCCCN(CCOc2ccc(Cl)cc2)C1 CC1(CN(C(C2(NC(C3CCCN3C3CC3)=O)CCC2)=O)C2CC2)CCCC1 Cn1[nH]c(C(=O)NC2CC2CNC(c2cnn(-c3ccccc3)n2)=O)nc1=O C1(C(=O)NCC(C)(C)OC(C)C)CC(C)CN(C(c2[nH]ccc2C2CC2)=O)C1 C=CCCCC(=O)N1CCCCC1C(N1CCN(C(C)(C)CC)CC1)=O C1(NC(CN(CCC)C)=O)C2CCN(C(c3ccc(O)c(CO)c3)=O)CCC12 C12(NC(c3c(CC)n[nH]c3)=O)CCCN(C(c3nc(C)oc3C)=O)CC1C2 C1(CC)(CC)CCN(C(=O)CC2CCN(CCSC)C2)CC1O C1(NC(C2CCC(CNC(c3cc(SC)oc3)=O)CC2)=O)CCCCC12CCC2 Cc1nc(CC(C)C)c(C(=O)NCC2(C(=O)NC(CN(C)C)C(C)(C)C)CC2)s1 c1(CC)nc(C(=O)NN(CCCC2CCC2)CCOCCO)c(Br)s1 CCC1=C(C(=O)N(C2CCCCC2NC(C2(C)CS(=O)(=O)C2)=O)C)CCCO1 C1(NC(C2(COC)CC2)=O)CCC12CCN(C(c1ccn3ccccc13)=O)CC2 C1(CN(C(CCCC#N)=O)C2CC3CC2CN3)CCCC2(CCC2)O1 c1(Cn2cc(CC(C)NC(=O)CS)nn2)ccc(F)cc1.c1(CO)cc(CO)on1 CC(CN=c1ncc([N+](=O)[O-])c[nH]1)NC(c1cccc(C(C)(C)C)n1)=O c1(C(N2C(CNC(c3cnco3)=O)CC2)=O)ccc2c(c1)CCC2 c1(CC)cccc2c(CNC3CC(CO)C4CC34)c[nH]c12 O=[N+]([O-])c1cccnc1S(=O)(=O)N1CCCC(n2ccnc2)C1 C1(C(N2CC(c3n(CC)cnn3)OCC2)=O)CC(C2CCCC2)C1 C(CCCOC)(C(=O)N(CCC(C)C)C)NC(C1C(C#C)C1)=O C1(NC(c2scc(CCOC)n2)c2nnnn2C2(C)CC2)CCC2(CCCC2)C1 C1(NC(C(C)NC(C(CC)SC)=O)=O)CCC(CC)CC1 C1(C(=O)NC(C2CC=CCC2)C(=O)NC23CCC(CC2)C3)CC(=O)NC(=O)N1 N1(c2c(Br)cnc(OC)n2)CCC(C2CC2)(CNC(=O)C(C)c2cccs2)C1 Cc1nc(N2CC=CC(NC(c3cc(O)no3)=O)C2)c(F)c(C)n1 C(CCCC(=O)N1CCC1CNC(c1ccc(C#N)o1)=O)N(C)C Nc1c(C(=O)NC2COCC2NC(C2CC(O)C2)=O)cccc1[N+](=O)[O-] N#Cc1c(Cl)cc(N2CCN3C(CCS3(=O)=O)C2)cc1[N+](=O)[O-] c1(C(COC)NC(=O)CC(=O)O)ccccc1F N1(C(CCCNC(C)=O)=O)C(C)C2CC1C2NC(=O)C=C1CCC(C)CC1 c1(C(=O)OC)nsc(=NCCC2CCCN(C(=O)CSC(F)F)C2)[nH]1 C1(C)(C(=O)NC(CN(C(CN(C)CC)=O)C)C)CC1(Cl)Cl C1(CNC(CSC(C)C)=O)CCN(C(=O)CN2CCCS2(=O)=O)CC1(F)F C(C(=O)N)N(C(=O)CN(C)CCOC)CCOC1(C(=O)OC)CC1.C=O C(=O)(CCCCC(C)(C)C)N(C)CC1(O)CCN(C(c2cc(Br)n[nH]2)=O)CC1 C1(CNC(C2C(CC)CCC2)=O)CC(F)(F)CN1C(=O)C(F)C(C)(C)O C12(C(=O)NC(C(C)C)(C)CNC(=O)CC(C)n3ccnc3)CCC(CC1)C2(C)C O=C(CCCn1cccc1)NC1COCC1NC(=O)Cc1cc[nH]n1 Cc1cc(C(=O)NC2CC2CNC(=O)CS(C)(=O)=O)cnc1C(F)(F)F C1(N(C(=O)CCSc2n[nH]c(O)n2)C)CCN(C(C2CC(F)(F)C2)=O)CC1 N1(C(c2ccc(C(N)=O)o2)C(=O)NCCCC)CC2C(C(=O)N(C)C)C2C1 N1(C(c2occ(C)c2)=O)CC(C2CCCN(C(C34CCC(C)(CO3)C4)=O)C2)C1 C12(NC(=O)Cc3cccnc3)CC3CCC(C1C2)N3C(c1cscc1C1CC1)=O c1(C(N2CCC(NC(C(C)N(C)C)=O)C2C)=O)cc2cc(Cl)ccc2o1 N1(C(N2CC(OC)C2)=O)CCOC(c2ccc(-c3cccc(F)c3)cc2)C1 C(C(=O)N(C1CN(C(c2ccncc2-n2cccn2)=O)CC1O)C)(C(C)C)SC c1(C2C(C3N(C(C)=O)CCCC3)C2)ccc(C)cc1-n1cc(CCC(=O)O)nn1 c1(OC)cc(OC)cc(CCC(N2CCC(C)(NC(c3ccon3)=O)C2)=O)c1 N1(C(C=CCOC)=O)CC(NC(c2cc(C(F)(F)F)cc(F)c2)=O)C2(CC2)C1 c1(C(N2CCC(CC=C)(NC(=O)C=CC3CCC3)CC2)=O)ccnc2ncnn12 CCC(CC)(C(=O)NC1CCC1C(N1CC(F)(F)C1C(C)C)=O)OC N1(C(C2CC(CC)(CC)C2)=O)CCC(C)(C)C(CNC(=O)CC2(C)CC2(F)F)C1 c1(C(N2CCCC(CNC(c3c(CC)c[nH]c3)=O)CC2)=O)cccc2oncc12 C(CC(=O)Nc1cc(CO)cc(F)c1)(C(F)(F)F)NC(C1(C#N)CC(=O)C1)=O N1(C(c2c(CC)c[nH]n2)=O)CC2CCC(C1)N(C(=O)Cc1ncoc1C)C2 C(=O)(CCCCC(C)=O)NC12CCCC(NC(CCNC(CC(C)C)=O)=O)(C1)C2 c1(C(=O)NC2C(C(=O)Nc3c(OCC)cccc3C)C2)ccc2ccnn2c1 N1(C(CC2(NC(C)=O)CC2)=O)CC(C(F)(F)F)OCC1C(=O)NCc1ncn(C)n1 N1(C(C)=O)CCN(C(=O)CN(C(=O)CCc2cc(C)no2)C)CC1 C(CC(C(=O)NCC(O)C1(Cl)CC1)NC(c1cncc(O)c1)=O)=CC N1(C(c2cn(CCNC(CNC(=O)OCC=C)=O)nn2)=O)CCOCC(O)C1 N1(C(C)=O)CC(NC(C2CCN(C(C3CN(C)C3)=O)CC2)=O)C(n2ccnn2)C1 C1(CCC(N2CCC(OCC)C2)=O)CCCN(C(c2cnc(C)s2)=O)C1 c1(N(CC=C)C)nc(N2CCC(C3CCCO3)C2)nc2scnc12 c1(CNC(C(C)C(C)(C)C)c2nnnn2C2(C)CC2)cc2cc(Br)cc(F)c2o1 N1(CCC(=O)NCCOCC)CCC(NC(C2CC(OCC)C2)=O)C1 Cc1n[nH]c(C)c1S(=O)(=O)NC1CN(Cc2ccn(C)n2)CC1C#N CC1=C(C(=O)N2CCCN(C(=O)C(c3ccccc3)F)CC2)COCC1 c1(OCC)ccc(N)c(C(=O)NC2CCCC(Nc3ncc(OC)cn3)C2)c1 c1(NC(CC2(NC(CC=CC)=O)CC2)=O)cccc(-n2cccc2)c1 c1(C(=O)NCC(C)N(C(c2cccc(N)n2)=O)CC)cc2sccc2s1 N1(C(C(C)N2CCCC2)=O)CC2CC(C1)N2C(C1CN2CCC1CC2)=O Cc1noc(C)c1CC(=O)NC1(CCNC(c2snnc2C2CC2)=O)CCC1 C=CCC(C)(C(=O)NCCC1CCCN(C(=O)CS(N)(=O)=O)C1)N(C)C c1(C(N2C3CN(C(c4c(C)nsc4)=O)C(C3)C2)=O)cc(F)c(Br)c(F)c1 C1(NC(c2cccc(SCC#C)c2)=O)CCSC12CN(C(C1CCC(O)C1)=O)C2 C(=O)(N=c1cc(SC)n(C)[nH]1)CC1(NC(C(CCC)N(C)C)=O)CCC1 c1(CC(=O)N(CC(CC)NC(=O)CCSC)C)csc(C(c2ccccc2)C)n1 C(=O)(C1=C(Cl)CCC(C)C1)NC(c1cccc(C)c1)CNC(C1(F)CC=CC1)=O c1(NCc2cn(CCN(C(c3c(C(C)C)onc3)=O)C)nn2)ccc(F)cc1 N1(C(C2CCC(OC)C2)=O)CC2CC(C(=O)NC(c3cncc(F)c3)C)(C2)C1 C1(C(N(C(C)CCNC(=O)Cc2ccccc2)C)=O)CCOCC12CCCC2 C1(NC(c2cc(OC)ns2)=O)CC2(C1)CC2NC(C1CCC2(CC2)C1)=O CC1(CCNCCc2nc(C3CC3)no2)CC(=O)C1 N1(C(c2c(CC)csc2)=O)CCC(C(=O)NCC2(C)CC2(C)C)CC1(C)C c1(C(=O)NC2CC(NC(CC=C)=O)C(O)C2)ccc(C)cc1Cl C=C(C)CC(C(=O)NC1CCC(NC(C2C(C)C2C)=O)CC1)NC(C)=O C1(NC(CC=CC)=O)CCCC(NC(c2csc(-c3ccc(F)cc3)n2)=O)C1 N1(C(=O)NC2CCC(CS(N)(=O)=O)C2)CC(C2CCCC2)C1 C12C3CN(CC13)C2=O.C1(NC(=O)CCOCC2CCCO2)CCC(CO)CC1 CCCCCCCC(O)C(F)(F)C(=O)N1CCCC1C1CCNC1=O Cc1nc(C(CO)NC(C2(C)CN(C(c3csnc3Cl)=O)C2)=O)n[nH]1 C(=O)(CCC(=O)NCC(c1cccc(Cl)c1)NC(C1CC(C)(O)C1)=O)OC C1(F)(CNC(C2C(c3n(C)cnc3)C2)=O)CCN(C(c2ccc(Cl)[nH]2)=O)CC1 C1(C(N2CCCC(N(C(C3C(C)SCCC3)=O)C)CC2)=O)CC2C=CC1C21CC1 C#CCC(C)(CC)C(=O)N1CC2C(C(=O)NCCCCCCCC)C2C1 C1(NC(C(C)C)=O)CN(C(c2cccc(-c3ccccc3F)c2)=O)CCC1F Cc1c(C(N2CCC(c3cnco3)C2)=O)oc(=O)c2ccccc12 N1(C(c2cncc(NC)c2)=O)CCN(C(=O)Cn2cnnc2)CC12CC2 C=CCC(CC(F)(F)F)NC(=O)Cc1csc(C2CC2)n1 C=CCC(CC(=O)NCCN1CC(C)(O)C1)NC(c1c[nH]nc1[N+](=O)[O-])=O N1(C(=O)C(C2CCOCC2)F)CCN(c2cc(F)ncn2)C(c2ccccn2)C1 C1(CNC(C(C)NC(CC)=O)=O)(COC)CCN(C(=O)C(C)SCC(C)C)CC1 c1(C(=O)NCC(CNC(c2c(C#C)c[nH]n2)=O)C)ccc(S(N)(=O)=O)s1 c1(C(=O)NC2C(C)CN(C(c3ccnc(C#N)c3)=O)C2)cc2cc(Cl)c(Cl)cc2[nH]1 Cc1cc(C(N2CC3C(NC(C4CC4C(C)C)=O)C3C2)=O)cc(C)c1 c1(NC(C2N(C(C3CCCN(C)C3)=O)CC(O)C2)=O)cc(Br)cc(Cl)c1O C(=O)(C1=CCN(C(=O)CC(=O)OC(C)(C)C)C1)NCC(C)O C1(NC(Cc2nc(C)oc2)=O)CCCC(NC(=O)CC2CCCN2C)C1 N1(C(CC(CC)C2CC2)=O)CCCC2CN(C(=O)Cc3c[nH]nc3O)CCC12 N1(C(C(CC)OCC)=O)CCC(CC)C1C(=O)N(C(CF)CF)C C(=O)(C(C)(C)CC(C)C)NCCN1CCN(C(C2CN(CC)C(=O)C2)=O)CC1 c12cnc3nccc(c3c1)[nH]c2=O.N1(C(C(C)OCC#C)=O)CC2C(C)C2C1 c1(NC(CN2CCC(NC(CC3C(C)C3)=O)C(O)C2)=O)ccc2c(c1)nnn2C c1(C(N2CC(c3n(C)ccn3)C(NC(=O)C(C)(C)F)C2)=O)cc(F)c(F)cc1N c1(NC)cnc(C(C)C)nc1C(=O)NC1CCC(NC(=O)CCCN(C)C)CC1 Nc1c(C(N2CCCC2CNC(=O)CCC2CCCOC2)=O)cccc1[N+](=O)[O-] c1(C(=O)NC(C(C)NC(c2cn(C(C)(C)C)cn2)=O)CO)ccc([N+](=O)[O-])n1C C(=O)(C(CCF)NC(=O)CC1CCCO1)N1CC(C)(CC=C)C1 C1(N(C(c2c(CC)scn2)=O)C)CCCN(C(=O)CC2(C)CCOC2)CC1 C(C(O)(C(F)(F)F)n1cccn1)N(CC(=O)NC(C)C)Cc1cccc(C)n1 c1(N(CC(C)NC(c2cnn(C(CC)CC)c2C)=O)C)cc(Cl)nc(C2CC2)n1 N1(C(C(CC)C2CCOCC2)=O)CCc2c(Cl)cc(F)cc2C1C.C1(N)CC(OC)C1 C1(NC(C2CC(=C)C2)=O)CC12CC(NC(c1n[nH]cc1Cl)=O)C2 C1(NC(C)=O)CCCCC1CNC(c1onc(-c2ccccc2)c1C(=O)O)=O c1(C(=O)NCCC(C)(C)NC(C2CCC(OC)C2)=O)cc(Cl)ncc1O CC(C(F)(F)F)(C1CCCC1)NCCCOc1ccccc1Br c1(C(=O)NC2(C)CN(C(C(CCC)N(C)C)=O)C2)cccn(C(=O)OC(C)C)c1=O C(C)(c1ccc(OC)cc1)=CC(=O)NC1CC(CNC(C(CCC)(C)O)=O)C1 C(=O)(C1Cc2ccc(C)cc21)N1CCC2(CN(C(c3c(CC)cccn3)=O)C2)C1 Cc1ccc(C(C)CC(N2CC(CNC(=O)CC#N)C(C)C2)=O)cc1 c1(C(N(C)CC2(NC(c3ccc(C(F)F)o3)=O)CC2)=O)nnn(C)c1N C1(CC=C)(C(=O)NC2(CO)CC3CCC2C3)CCCNCC1 c1(CNC2(CCC)CCOC2)cc(OCCO)cc(Br)c1 c1(C(=O)NCC2CN(C(c3ccc(Cl)o3)=O)CCO2)ccnc(Cl)c1F C1(CC)CN(C(=O)C(C)(C)C(C)NC(C2CCN(C(N)=O)CC2)=O)CCCO1 c1(C(=O)NC(C(=O)NCC(CC)(C)CO)C)c(C)[nH]c(C)c1C N1(CC(N2CC(C)N(C(C3CN(CP(C)(C)=O)C3)=O)CC2)=O)CCc2sccc2C1 c1(CNC(C2=C(C)OCC2)=O)cnn2cccc2c1Cl c1(CC(=O)OCC)nc(CC(=O)C(Cn2cc(C)cn2)SC)no1.NC CC(C)(CC(=O)NCC1C2CN(C(c3ccc(CO)cc3)=O)CC12)CC(F)(F)F c1(C(=O)NC(CCNC(C(CC)NC(N)=O)=O)C)cc(Br)cc2c1OCC2 C1(NCC2CN(C(C(CC)C)=O)C2)CC2(CCC2)CCN1C(=O)OC(C)(C)C c1(OC)cc(C(=O)NCc2ccccc2Br)cnc1-c1ccccc1NC(N)=O N1(C(c2onc(C)n2)=O)CCN(C(C2CCCN(CC3CC3)C2)=O)C(C(C)C)C1 C1(NC(Cc2ncc(C)s2)=O)CCCC(NC(=O)CN(c2ccncc2)C)CC1 C12COCCN1NC(=O)C2.C(C)(C)(C)OC(N(CCN(C)C)CCF)=O C1(CN(C(=O)C(c2ccccn2)O)C)CCN(C(CCCN(C)C)=O)CC1 CCCCCCC(C)C(=O)N(C1CCCC1)CCNC(c1snc(Cl)c1Cl)=O N1(C(C2N(C(=O)NC)CCC2)=O)CCN(C(c2coc(CC)n2)=O)C2(CCC2)C1 C1(C)(CNC(C2C(CCC)C2)=O)CCCN(C(c2cc3sccc3s2)=O)C1 N1(C(c2cnc(OCC)s2)=O)CCN(C(C23CC2COC3(C)C)=O)C(C)C1 C#CC1(C)CCCN(C(C2CCC(NC(=O)C#CC3(C)COC3)C2)=O)C1 c1(C(=O)NC2CC(CNC(c3c(CCC)nco3)=O)C2)cc(N)cc([N+](=O)[O-])c1 N1(Cc2c(C)ccc(Cl)c2)CC(C(=O)N(C)C)c2cc(Br)ccc21 CCCCC(F)C(=O)NCCn1cnc(C(N2Cc3ncsc3C2)=O)c1 C1(CNC(C(CC)(F)F)=O)CN(C(c2cccc(C3(C)CC3)c2)=O)CC12CC2 N1(C(c2sccc2Cl)=O)CCC(N(C(=O)CCc2ccccc2)CCO)CC1 N1(C(C2C(c3ccc(C)cc3)C2)=O)CC2(CC(NC(C3(CF)CCC3)=O)CO2)C1 C1(O)(CN(C)C(C2CC2F)=O)CCCN(C(c2cccc(-c3ccsc3)c2)=O)C1 C(CN=C(NC1CCC1)N1CCC(OC(C)C)C1)NC(=O)NCC(N)=O C(CNC(c1c[nH]nc1Cl)=O)(CCNC(=O)CC1CCC2CC12)OC Cc1nn(C)c(F)c1C(=O)NC(C1CCCN(C(c2ccn(C)c2)=O)C1)C C(=O)(C(C)C(C)O)NC(C)CNC(C1(C)CC1C(F)(F)F)=O c1(C(N2CC(NC(COC)=O)C3(C2)CC3)=O)ncc2ccccc2c1O Cc1cc(C(=O)N(CCCC(=O)N(C)CC2(C)CCC2)C)c[nH]c1=N C1(NC(C(N)=O)=O)C=CC(CC(=O)NCCCSC(F)F)C1 c1(CC(=O)NC2CN(C(C=CC(=O)OCC)=O)CC2C)ccc(F)c(Cl)c1F c1(C(=O)NCC(=C)CCNC(=O)CC2(O)CCCOC2)c(Br)ccc(C)c1F C1(NC(C)=O)CCCN(C(=O)C(=O)NCCSCC2CC(C)CO2)C1 c1(NC(C(n2cc(C(=O)NC3C(C)(C)C3(C)C)nn2)C)=O)cc(Cl)c(Cl)c(Cl)c1 CC1CC(NC(=O)CC(=O)OC(C)(C)C)CN(C(N)=O)C1.C12CN(CC1C)C2=O Cc1cc(C(=O)NCC(CNC(C2CCn3ncnc3C2)=O)CO)c(Cl)cc1F Cc1c(Br)sc2ccccc12.C(C)(CC(C)C)OCCC(=O)N(C)CCN(C)CC C1(C(=O)NC(C(C)O)C(=O)NC(C)Cc2cnn(C)c2)CC2CCC1CC2 C12(C(=O)NCC3(NC(=O)NCC)CCCC3)CCCC(CN1C(=O)C(C)CF)C2 c1(NC(C2N(C(c3ccc(C)cn3)=O)CC(O)C2)=O)c(Cl)c(F)nc(F)c1Cl N1(C(COCC)=O)CC2(CCC2)CC1CNC(C1C(C)(C)OC1(C)C)=O C(C(F)(F)C(C)(C)C)N(c1ccnn1C)C(=O)NC(CC#C)CC=C N1(C(C)C)CCOC(C(=O)NCC(C(C)C)NC(=O)Cc2ccns2)C1 c1(OC)cc(N)c(C(=O)NC2CCCC(NC(=O)C3=COCCO3)C2)cc1OC c1(C(CC(=O)NC(CC(=O)OC)C)C)cccc(C)c1 c1(CCC)cc(C(N2CCCC2CN(C)C(C2CCC2C(F)(F)F)=O)=O)c(C)o1 CC1CC(NC(C2CC(=O)N(O)C2)=O)CN(C(=O)Cc2cccc(Cl)c2)C1 C1(NC(CC(C)CF)=O)CN(C(C2CC(C)(C)CO2)=O)CC1(C)C c1(CC)ccc(C(N2CCC(C(=O)N(C3CCN(C(C)C)C3)C)(CC)C2)=O)cc1 Cc1ccnnc1C(=O)NC1CC(CNC(=O)CCN2CCCCC2)C1 c1(C(=O)NC(C2(O)CN(C(c3sc(CC)c(C)c3)=O)C2)C)ccc2ccnn2c1 N1(C(=O)NC(c2nc(C)c(N(C)C)s2)C)CC2(CCN(C(=O)OC(C)(C)C)C2)C1 C1(NC(N2CC3CCC(C2)N3C(=O)C2=NOCC2)=O)COc2ccccc2O1 c1(C(=O)NCc2c(C(=O)NC(C#C)C(C)OC)occ2)nc(C)sc1C N1(C(c2c(CNC(CC3CCCC(C)O3)=O)occ2)=O)CCC12CCC(C)CC2 c1(C(N(C2CCCN(C(CC(=O)OCC)=O)CC2)C)=O)cc(F)c2[nH]nnc2c1 c1(C(=O)NC(C)CCCNC(=O)Cn2ccnn2)ccc(C(F)F)c(F)c1 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(NC(C2CC2C)=O)CC2(CCOCC2)C1 CC1=C(C(=O)NC2CCC(NC(=O)C(C)(C)N(C)C)C2)CCO1 c1(C(N(C)CC2N(C(c3cncc(C)n3)=O)CC(F)C2)=O)c[nH]c2ncccc12 S(=O)(=O)(c1cn(C)cn1)NCC(N1CCC(N(C(C(CC)SC)=O)CC)C1)=O c1(C(N2CCC(N(CCC)C(C3CC3F)=O)C2)=O)cc(Br)c(C)cc1F Cc1cc(C)c(C(=O)NCC2(CNC(C3(O)CCOCC3)=O)CCCC2)c(=O)o1 N1(C(C(C)=C(CC)C)=O)CCC(CNC(=O)COC2CC2(F)F)C(F)(F)CC1 c1(C(=O)NC2CN(C(c3n[nH]c(C)c3F)=O)C(C)C2)c[nH]c(=O)c2ccncc12 N1(C(C(C(=O)OC)OC)=O)CCC2CC2(NC(=O)CCNC(C)=O)CC1 Cc1cccc(-n2cc(C(N3CC(N(C)C(C4CCC(C)(C)C4)=O)C3)=O)nn2)c1 C1(NCc2cn(Cc3snc(C(=O)OC)c3Br)nn2)CC(C)(C)C(=O)O1 C1(C2CCN(C(=O)CSCc3ncc[nH]3)CC2)(NC(CC(COC)C)=O)CC1 c1(NC(C2N(Cc3nccc(C)c3)CCCC2)=O)ccc(F)c(Br)c1F CCCC(C(=O)N1CCC1CNC(C1(CCOCCOC)CCC1)=O)C(C)C C(C)(C(C)(C)CN(C(c1ccc(Cl)o1)=O)C1CC1)NC(C)=O C1(NC(c2nc(OCC)sn2)=O)CCCC(CNC(c2c(C)csc2Cl)=O)C1 c1(OC)ccc(C(O)C(=O)NCCC(C)N(C)C(c2cnoc2C2CC2)=O)cc1 N1(C(c2c(C)cc(C)nc2)=O)CCC2C(CCN2C(=O)CC2CCOC2)C1 C=CCCCC(C(=O)NCCOCCN(C)C)NC(c1cnc(Cl)n1C)=O C(C(C(=O)N1CC=CC1CF)NC(=O)CC1CCC(=O)N1)SCC C=C1COCCN(C(=O)C2=CCN(C(=O)CC(C)(C)C)C2)C1 CCCC(C(=O)NC1CC(CNC(C2(C(=O)N(C)C)CC2)=O)C1)OC C1(C(=O)NCC2(NC(CCC=C=C)=O)CCOC2)COc2cc(OC)ccc2C1 C1(N(C(COCC(=C)C)=O)C)CCN(C(c2nccn3nccc23)=O)CC12CC2 c1(OCC)cccnc1C(=O)NCC1(F)CC(CNC(C23CCC(CC2)C3)=O)C1 N1(C(C2ON=C(C(C)C)C2)=O)CCC(C2CCN(C(=O)CCC3CCC3)C2)CC1 c1(C(=O)NC2OCC(=O)N(C)C2c2cccnc2)c[nH]c2c(F)ccc(F)c2c1=O c1(C(c2nnnn2CCC2CC2)NCC(Cl)(Cl)Cl)ncccc1Cl c1(CC(C(=O)NC2CC(F)(CNC(Cc3c(C)ocn3)=O)C2)C)cccc(F)c1 c1(OC)ccc2c(C(=O)NCC3(O)CC(NC(=O)CCCF)C3)ccnc2c1 c1(C(N2CC(OC)C(NC(c3ncc(C)cc3F)=O)C2)=O)c(F)ccc(Cl)c1F c1(C(=O)NCC(CC)NC(C2CC(C)C2(C)C)=O)cnc(OC)nc1 C1(C(C)C)CN(C(C2C=CCN(C(=O)CC(Cl)Cl)C2)=O)CC(=O)N1 N1(C(Cc2n(C)nnc2)=O)CC(NC(c2cc3cccnc3[nH]2)=O)C2(CCCC2)C1 c12cc3c([nH]1)CCN(C3)Cc1c-2cccc1F.C(=O)(CN)OC c1(CC(N2CCC(NC(c3c(C)cns3)=O)C(CO)C2)=O)ccc2c(c1)OCO2 C(CC(=O)N1CCC(CCNC(=O)CSc2n[nH]c(=N)s2)C1)(C(F)(F)F)OC C12(NC(C=CCOC)=O)CCC(CN(C(=O)CCCCNC(C)=O)C1)C2 c1(OC)ccc2c(c1)CC(C(C)OC)CN2C(=O)NC1(c2ccccc2F)CC1 C1(C(=O)NC(c2c(C)occ2)=O)CCCN(Cc2ccc(C3CCC3)cc2)C1 n1(C(=O)OC)cc(CNc2cc(C)ncn2)c(C)n1.C12CCC(CC1)N2 CCC(O)C(F)(F)C(=O)N1CCC(NC(c2nc(Cl)sc2Cl)=O)C1 C1(F)(CNC(CC2CC(OC)C2)=O)CC(NC(=O)CCCC2CCCO2)C1 O=C(CCS(=O)(=O)C(F)(F)F)NC1CC(O)CN(C(c2ccsn2)=O)C1 Cc1cc(CNC(C2CCCCN(C(=O)CC3C=CCCC3)C2)=O)cc(C)n1 n1(CC(N2CC3C(NC(N4CCC(C)(C(N)=O)C4)=O)C3C2)=O)ncc(C#N)c1N N1(C(c2c(C)oc(Cl)n2)=O)CC(C2CC2)(C(=O)NCC2(C)CCCCO2)C1 C(C)(C)(CC(=O)NCC(=C1CN(C(c2cnn(C)n2)=O)C1)F)OC C1(C(NOCCCC(=O)OC)=O)(NC(C2CC(F)C(=O)N2)=O)CCN(C)C1 c1(C(N2CCC(CNC(C3CC3(Cl)Cl)=O)C23CC3)=O)ccnc2ncccc12 CC1(C)CN(C(C2CC3CCC2CC3)=O)CCC1C(=O)NCCN1CCOCC1 Cc1nc2cc(C(=O)NC3CC(O)CN(C(c4cnns4)=O)C3)ccc2s1 C1(C(=O)NCC(c2cnn(C)c2)C)CC2CC1CC2NC(c1cc(Cl)cs1)=O C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCC12N(C(COCC=C)=O)CCC1CC2 C1(CNC(c2c(N)sc(C)c2C)=O)CC2CC(C1)N(C(=O)C=CCO)C2 O=C(CC1=CSC2=NCCN12)NCC(C1CC1)NC(C1CCC2CCCCN12)=O C1(C(=O)NCCCN(C(=O)C(O)C(C)C)CCC)CCC(C)(C)CO1 Cc1ncc(S(=O)(=O)NCC2(c3cc(F)ccc3C(F)(F)F)CCCC2)o1 N1(C(=O)C=CCn2cncn2)CCCC(NC(C2(CO)CCOCC2)=O)C1 CC(C)CCC(F)C(=O)NC1CC2(C1)CC(C(=O)NC1COC(C3CC3)C1)C2 N1(C(CC(CCCC)NC(=O)Cc2cc(C)on2)=O)CCC2CN(C)CCC12 CC(C)C(C#N)C(=O)NCC1CCCCN(C(c2ccsc2)=O)C1 c1(OC)cc(OC)c(C(N2CCCCC(NC(C3CCOC3C)=O)C2)=O)cc1N CC1CCc2c(C(N3CC(O)(CCNC(=O)CCn4ccnc4)C3)=O)csc2C1 N1(C(C2C(=C)C2)=O)CCCC2C1CCCCN2C(=O)CC=CC(C)(C)C c1(C(=O)NC2C(NC(C3(N4C(=O)COCC4)CC3)=O)C2)cnn2ncccc12 C(=O)(CCCC(C)(C)C)N1C(C)CN(C(=O)C(C)(C)C=CCF)CCC1 N1(C(c2cc(CC)ncc2)=O)CCCC(C2CCN(C(C3(C)COC3)=O)CC2)C1 c1(CC(=O)N(C(CN(C(C=CCOC)=O)C)C)C)c(OC(C)C)cccc1Cl c1(NC(=O)NCC(COC)COC)nnc2n1CCC2.c12cc(on1)C1(CC1)C2 C1(C(N2C(CN(C(CCC(=O)NCC)=O)C)CCC2)=O)CC2C(C1)C2(C)C c1(C(=O)NC2CC(C)N(C(C3COC(=O)N3)=O)CC2)cccn2nncc12 N1(C(CCCSC)=O)CCC(NC(C2(F)CC2c2ccccc2)=O)CC1 c1(C(N(C2CC(C(N(CC#C)CC)=O)C2)C)=O)ncoc1C C1(OCCC)CCCN(C(C2(NC(=O)CCCN(C)C)CCSC2)=O)C1 C12(C(=O)NCCCCNC(c3c[nH]nc3OCCF)=O)CCC(N(C)C)(CC1)C2 c1(C(N2C(CNC(C(n3ccc(C)n3)C)=O)CCCC2)=O)cccc([N+](=O)[O-])c1 C(=O)(C1=COCCC1)NCCNc1cc(OC(C)C)ncn1 N1(C(C(c2cccc(C)c2)=O)=O)CC(NC(=O)CCC(N)=O)CC(C)(C)C1 C1(CN(C)C(c2c[nH]nc2-c2ccn(C)n2)=O)CN(C(C2(Cl)CC2)=O)CCO1 C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)CC2CCC(C)(O)CC2)C2(CCCC2)C1 C(C1CCCC1)=C(C)C(=O)NCC(C1CCOC1)NC(=O)CCCc1ncco1 c1(COC(c2c(CC)cco2)=O)c(F)cccc1Br N1(C(COCP(C)(C)=O)=O)CCC2CCC(C1)N2C(=O)CCc1ncccn1 C1(C=O)CCC2CN(C(=O)CN3CCn4ccnc4C3)CC12.c1(CC)ncc(C)s1 Cc1c(C(F)(F)F)cccc1C(F)(F)F.C(=O)(C(F)F)N(CC(C)C)C C1(C(N2C(C)(C(=O)NCC(COC)(C)C)C=CC2)=O)CC(C)CC(C)C1 C(CC(=O)NCC1CCN1CCCO)OCC(N)=O C1(C(c2c(OC)cccc2)NCCCCCCO)CC2CC1CC2(F)F c1(C(=O)OCc2n(C)nc(C(F)(F)F)n2)cc(F)c(Cl)cc1[N+](=O)[O-] Cc1cncc(CC(=O)NCCCCCN(C)C(C2CCC(C)C2)=O)c1 C(C)(C)(C(C)CC(=O)N(C(C)COC)C)NC(CC(C)OCC)=O C1(NC(C(C=C)OC)=O)CCN(C(c2sc(C(C)C)nc2C)=O)C(C)C1 CCC(C)(C#N)C(=O)N1CC(C(=O)NCCOCCSCCO)C1 Cc1ccc(C)c(C(=O)NCC2C3CC2N(C(=O)C(c2ccccc2)F)C3)c1 Cc1cc(F)ncc1C(=O)NCC1(O)CCN(C(=O)C(C2CCC(=O)N2)C)CC1 C1(NC(COCC)=O)CCCN(C(c2ccc(COC)cc2F)=O)CC1 Cc1nc(CNC(=O)CCNC(N)=O)oc1C(=O)N(C)CC1OCCC1(C)C N1(C(C2C(OC)(OC)CC2)=O)CCCC(C(=O)Nc2cn(C)c(O)n2)C1 CC1(C)CCC(C(=O)NCCCC2CCOCC2)CN1C(c1cccs1)=O CN1CCN(C(c2ccc(C(F)F)s2)=O)CC1CNC(c1ccncc1F)=O c1(C(N2CC(F)CC(NC(c3cccc(C)c3)=O)C2)=O)ccc2c(c1)nnn2C C1(C(N2CCC(NC(CN(CCC#C)C)=O)C2C)=O)Cc2nccnc2C1 C(=O)(N=c1cc[nH]cc1F)C1CCN(C(C(C)(C)CCl)=O)CC1 S(=O)(=O)(CCC(=O)NCC(O)CNC(=O)CCS(C)(=O)=O)N(C)C c1(CC(=O)N(CCCNC(C2(CC#C)CCOC2)=O)CCOC)cc(C)cc(C)c1 C(=O)(C(C(C)C)C1CCCCC1)NCC(COC)(C)O C1(CC(=O)NC(c2cn(CCOC(C)=O)nn2)(C)C)CC2C=CC1C2 C1(OC)CC(CNC(=O)CCn2ccnc2)N(C(c2oc(C(C)C)nc2C)=O)C1 C(N=c1nnc(C)c(C)[nH]1)c1ccc(CNC(C(=C(C)C2CC2)F)=O)c(F)c1 C1(C(N2CC(C)C(CNC(=O)C3=CCCCO3)CC2)=O)Cc2cc(F)ccc2O1 C1(NC(CCC#C)=O)CCN(C(C2CCC(CC)O2)=O)CC1F C1(OC)CN(C(=O)Cn2ncccc2=O)CC1NC(=O)C=C1CCCCC1 C(C(=O)NC)(C(CC(C)C)OC)N1CCCN(NC(=O)OCCOCC)CC1 C(=O)(CC(C(F)F)N1CCOCC1)N(CC)CC1CCCN1C(=O)C(C)OC c1(CSCCNS(=O)(=O)CC2CCOC2)cc(Cl)ccc1Br N1(C(C(CSC)O)=O)CCC(C(C)NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CC1 N1(C(CC=CCNC(C(C=C)(C)C)=O)=O)CCOCC(C)(F)C1 C1(C(CNC(C(C=CC)O)=O)F)CCN(C(C2(Sc3ccccc3)CC2)=O)CC1 Cc1cc(C(=O)NC2CCCC2C(=O)Nc2cc(Cl)ccc2F)nc(Cl)c1 N1(C(C(=O)NCC(CCC)(C)C)=O)CCOC(COC)C1 C1(C(=O)NC(CCNC(CCC#C)=O)(C)C)CCC(C)(C)CC1 c1(CC)cccc(C(N2CCC(NC(c3c[nH]nc3C(F)F)=O)C(C)C2)=O)c1N c1(C(=O)NCC2C3(CCN(C(CCC=C)=O)CC3)C2)cc(S(N)(=O)=O)sc1C C1(N)CC1C1(C)COC1.C1(C(C)C)CC(OC(F)(F)F)CCO1 N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(c1ccc(CO)o1)=O)C2 C1(OC)CC(N=c2[nH]c3c(c(=NCCOCCO)[nH]2)CCC3)C1 c1(C(=O)NCCCCNC(C(C(C)O)NC(=O)C2CC2)=O)ccc(S(C)(=O)=O)s1 Cc1cccc(C(N2CCOCC2C(=O)N(C(CCO)C2CC2)C2CCC2)=O)n1 c1(CCNC(=O)NC(c2cnnn2C)C)cccc2c1OCCO2 C1(CNC(C=CCC)=O)CCC12CCN(C(=O)CN(S(C)(=O)=O)C)CC2.NC C12(CNC(CCCC(N)=O)=O)CC(CCO1)N(C(C1CC(C3CCC3)C1)=O)C2 c1(C(=O)N(C2CCN(C(=O)CC3CC3)C2)CCO)ccc2c(n1)NCCO2 Cc1nnc2n1CC(C(=O)NCC1(C)CC(NC(c3ncccc3F)=O)C1)C2 n1(CCC(=O)NC2(CCNC(C(C=C)(C)O)=O)CCC2)cc[nH]c(=O)c1=O CC1CC(C(N2CCCCC2C2(NC(=O)CSC3CC3)CC2)=O)CC(C)O1 C1(NC(c2cccnc2)=O)CCNCCC1c1ccccc1.c1(N)ccccn1 C1(c2n(CC)cnn2)CCN(N2CC3(CCC4(CC3)OC4)C2)C1 N1(C(C2(COC)CCCO2)=O)CCN(C(C2CC(C)OC2C)=O)C(C)C1 N1(C(c2cccc(OCC)c2)=O)CC2(C1)SCCC2NC(=O)CC1CCC2CC12 C1(C)(C(=O)OC)CC2(CC(NC(=O)NC(C)C(N3CCSCC3)C)C2)C1 N1(C(=O)NCC2CCN(C(C)C)C2)CCC(O)(c2cccc(Br)c2)CC1 N1(C(c2nc(SC)sc2)=O)CCCCC1C(C)NC(c1ccc(C(N)=O)o1)=O c1(C(=O)NCc2ccc(I)c(C(F)(F)F)c2)c(O)ccc(F)c1F CCC(C)(CNC(=O)C(F)C(C)(C)O)C(=O)N(C1(COC)CC1)C N1(C(c2ccc(OCOC)cc2)=O)CCn2ncnc2C1.C1(CO)(O)CCOC1 c1(C(N2CC3CCC3(C(=O)Nc3cccc(Br)n3)C2)=O)nc2ccccc2[nH]1 C1(CNC(c2cc(COC)[nH]n2)=O)CC(C)CCN1C(c1[nH]c(C)nc1C)=O CC1C2CCCCC2CN1C(C1(C(C)NC(=O)CC2CCCCO2)CC1)=O c1(C(C)=O)cc(C(=O)NCC(C)N(C(=O)C(c2nc(C)cs2)C)C)cnc1C C(=O)(CCC(=O)N1CCOC(CN(C(=O)C=Cc2nccs2)C)C1)NCCC C(C1=CCCOC1)N(C(CNC(CNC(CCC)=O)=O)=O)C C1(NC(c2nc(C(C)NC(C3(CC(N)=O)CC3)=O)oc2)=O)CCCN(O)C1=O C1(C(=O)NCC(C)(C)NC(C(COC)C)=O)CC2(CCC2OC)C1 C1(N=c2ncnc(NC)[nH]2)(C(=O)Nc2c(C)cccc2)COC1(C)C c1(C(N2C(C(=O)Nc3cc(CO)nc(Cl)c3)CC2)=O)cccc2c(O)cccc12 c1(OCC(CN(C)NCc2ccc(OC(F)F)cc2)O)cc(O)c2ccoc2c1 c1(Cn2cc(CNC(=O)CCOc3ccc(F)cc3)nn2)c(Br)cccc1Br c1(-c2c(OC)ccc(C)c2)nc(C2CCCn3ccnc32)n(C(C)C(C)C)n1 C#CCC(C)C(=O)NCC1(F)CC(CNC(C2CC2(Cl)C(=O)OC)=O)C1 c1(CCCC(=O)NC(C)CC(C)NC(=O)C=CCN2CCCC2)c(F)cccc1F C(=O)(CCCCC(C)C)N1CC(CC(=O)NC(C)Cn2ccnc2)OCC1 N1(C(C(C2CC2)OC)=O)CCCC1CN(C(=O)C(=O)N(C)C)CC1CC1 C1(NC(=O)NCC23CCC(C(=O)OC)(C2)CO3)CC2(CCC2)C(=O)O1 Nc1ccc(C(=O)NC2CN(C(C3(Br)CC34CCC4)=O)C2)c([N+](=O)[O-])c1 c1(C(C)CC(=O)NCCOC2CN(C(=O)C=C3CCOCC3)C2)cccc(F)c1 c1(CC(=O)NCC2C(NC(CCc3cc(C)on3)=O)C2)cccc2nonc12 Cc1cc(C=CC(=O)NC2CC23CC(NC(=O)C(F)=CC2CC2)C3)ccc1F n1(CC(=O)NCC2C(NC(COCCOC)=O)C2)ncn2cccc2c1=O C1(NC(CN(c2ccncc2)C)=O)CN(C(=O)CCC2CC2(F)F)CC1C(F)F c1(CC)cncc(C(N2CC3C(CN(C)C(C4CC5CCC4O5)=O)C3C2)=O)n1 C1(C(N2CCC(OCCNC(CCCCSC)=O)C2)=O)CCC(O)CN1C c1(C)cc2n(n1)CCC2.N1(CC)CCOCC1C1(C)CC1 C(C(O)C(=O)NCC(C)(C)OCCNC(=O)Cc1cc(C2CC2)on1)=CC C1(C(=O)NCCc2cn(CC)nn2)(CF)CCN(C(C2COCCO2)=O)C1 N1(C(CCc2ccc(C(=O)OC)o2)=O)CCCC1C1CCCO1 Cc1cncc(C=CC(=O)NC(C)(CNC(=O)C=Cc2csc(C)n2)C2CC2)c1 C(C)(N=c1[nH]c(CO)nc2c(C)csc12)C1CN(CC2(C(=O)OC)CCCO2)C1 c1(CN(C=O)Cc2n(CC(C)C)ncc2)cc(C#N)ccc1F C(CC(O)CC(=O)NCc1csc(=NC)[nH]1)SC.C12CC3(CC3)CN1C2 c1(C(=O)NCC(C)CNC(C2COC(=O)O2)=O)ncc2[nH]ncc2n1 c1(C(N(CCNC(C2C(C(=O)OC)CCO2)=O)C(C)C)=O)cc(O)cc(O)n1 N1(C(=O)OC(C)(C)C)CCOC(C)(CC(=O)NCCSc2cocc2C(=O)O)C1 c1(C(C(=O)N(CCNC(C(CSC)C)=O)C(C)C)(F)F)ccccc1C#N C(CCC(O)C(=O)NCC1CN(C(C)C)C1)NC(C1CC(F)C1)=O c1(C(N2CCC3C(NC(C(C)(C)C)=O)C32)=O)cc(C(F)(F)F)c(Cl)cn1 CC1CN(C(c2ccc(O)cn2)=O)CC1NC(=O)C(C)(C)c1ccsc1 c1(NC(N2CN(CC)C(=O)C2)=O)nc(Cl)nc2c1c(O)nc(=O)n2CC#N C(C(C)CS(=O)(=O)NC(C)C(C)n1cncn1)OCC C12(C(=O)NC3CC4CN(C(=O)CC(F)(F)F)C(C3)C4)CC(CO)(C1)OC21COC1 N1(C(c2ccc(CC)cn2)=O)CC2CC(C1)N(C(c1nc3cccnc3s1)=O)C2 S(=O)(=O)(c1cnccc1C(=O)N(C)C)N1CCC(NC(C)=O)C1 Cc1cc(C(=O)NCC2C(C)CCN2C(=O)CC2(C#N)CC2)c(O)c(C)c1 c1(C(=O)NC2(CCCNC(C(C3CCOCC3)C)=O)CC2)ccc(CO)c(F)c1 C1(CC=C)(NC(=O)C(C)c2ccsc2)CCN(C(C2CC(F)(CO)C2)=O)C1 Cc1cnn(C)c1C(=O)NCCCC(C)NC(c1cncnc1C)=O Cc1ccc(C(N2CC=CCC2C(=O)NCC2(CO)CC3CC3C2)=O)c(O)n1 Cc1nn(C)c(C)c1S(=O)(=O)N(c1ccc2ncnc(O)c2c1)C1CC2CNC1C2 Cc1ccc2ccc(C(=O)NCC3(CNC(c4cnoc4)=O)CCCC3)nc2c1 c1(C(N2CCCC(CCCCNC(CCCOCC)=O)C2)=O)cc(C)ccc1N N1(C(C(C2CN(C(=O)C3=CCSC3)C2)OC)=O)CCC12CCCOCC2 c1(OC)c(C(N2CC(CC(C)NC(=O)CC3CCC(C)CO3)C2)=O)csc1C C(=O)(CC(C(F)F)NC(c1ccc(F)cc1C)=O)NCC(C(=O)OCC)(C)O N1(C(c2cc(CCC)nc(O)c2)=O)CC2CCN(C(c3cncn3C)=O)CC2C1 C1(C(N(CC(C)C#N)C)=O)CC(O)CCN1C(=O)C(C1CCOCC1)C n1(CC)c(C)cc(C(N2CCN(C(=O)CCc3cn[nH]c3)CC2C2CC2)=O)c1C c1(CNC(C(C)n2ccnn2)=O)nc(C(=O)NC(C)(C)CC2CCC2)co1 C(C(C(=O)NC1CCCSC1)C(C)(C)C)NC(CC1ON=C(C)C1)=O N1(CCC)CCCC1C(N1CCC(CNC(=O)CCN(CC(F)(F)F)C)C1)=O c1(C(N2C(C(C)NC(C(CC=CC)C)=O)CCC2)=O)cc(OC)cc[n+]1[O-] C1(C(=O)NCCCNC(C2C3COCC23)=O)CCN(C(=O)NC2CCC2)CC1 C(=O)(CCCCC(F)(F)F)N(CC(O)CN(C)C(c1csc2c1CCCC2)=O)C c1(C(N2CCCC(C(C)NC(CCC(=C)Cl)=O)C2)=O)ccc(N)c([N+](=O)[O-])c1 C#Cc1cnn(CC(=O)N(C(C)CNC(C2CC2C#N)=O)C)c1 c1(C(N(CC(C)OC)CC)=O)cnc(O)c(C)c1.C12(CCCC1)CCC(=O)N2CC c1(C(N2CCC(NC(c3c(COC)cccc3)=O)C2C)=O)cc(OC)nc(C)c1 CC(C)CC(CC(=O)NC1CCCN(c2ccccc2)C1)CC(N)=O C1(CNC(C2N(CC)C(=O)CC2)=O)CCN(C(c2csc(COC)n2)=O)C12CC2 C1(O)(CCNC(=O)Cc2ccc(Cl)cc2)CCCN(C(=O)C=CCF)C1 C(C(CNC(c1cn(CCF)nn1)=O)CO)NC(CCNS(CC)(=O)=O)=O CC1=NOC(C(=O)NCC2CCN2C(c2ccccc2C(N)=O)=O)C1C C1(C(=O)NC2CCN(C(c3ncccn3)C)CC2O)Cc2cccnc2C1 C1(NC(Cc2cccc(C)c2Cl)=O)CCCN(C(c2cc(O)cc(Cl)c2)=O)CCC1 Cc1ccc(C(N2CC(C)CCC2c2cccc(CO)c2)=O)cc1S(=O)(=O)C(C)C O(NC(=O)C(CSC1(C)CCCC(=O)N1)NC(=O)OC(C)(C)C)C(C)(C)C c1(C(=O)NCCC2CCCN(C(CC(C)C(F)F)=O)C2)c[nH]c(=O)c2ccnn12 C(=O)(N=c1nc(OCc2ccccc2)[nH]n1C)C1C2(C)C(C)(CSC2)C1 Cc1sc(C(=O)NCC2CCN2C(c2cccnn2)=O)c(Br)c1C c1(C(=O)NCC(C2CCCC2)NC(c2cc(COC)on2)=O)cc(C)cnc1F C(=O)(C(C)(C)n1cnnn1)NCCN(C)C(C1CC1F)=O N1(C(c2c(O)ccc(C)n2)=O)CCCN(C(c2cncc(C)c2Cl)=O)CC1C CC(C)C(C)(CNC(=O)Cc1cccnc1Cl)NC(c1csc(C(F)(F)F)n1)=O c1(C(=O)NC2CN(C(c3c(C)ocn3)=O)CC(C)(C)C2)ccn2c(O)nnc2c1 n1(C(C(=O)NCCN(C(c2c(C)nc(O)[nH]2)=O)C2CC2)C)nc([N+](=O)[O-])cc1C Cc1cc(C(=O)NCCCN(C(C2CCC(=O)C2)=O)C2CC2)nc(O)n1 N1(C(c2cc(C)n(C(C)C)n2)=O)CCCCC(NC(=O)CC(C)C(C)C)CC1 C1(CC#C)CN(Cc2c[nH]nc2-c2ccncc2)C12CCC2 c1(NC)cc(=O)n2oc(C)cc2n1.N12CCC(CC1)N(CCO)C(CC)C2=O Cc1cccc(C(N2CCC(C)(NC(c3cc(-c4cnn(C)c4)[nH]n3)=O)C2)=O)c1 C1(S(N)(=O)=O)(C(=O)NC2C3CC(NC(Cc4c(C)noc4C)=O)CC32)CCC1 N1(C(c2cccc(C)c2I)=O)CC23CCCCC2(C1)CN(C(c1cc[nH]n1)=O)C3 c1(C(=O)NC(C2OCCN(C(CC(=O)NCC)=O)C2)C)cc(C)cc(C)n1 c1(NC(C2(C)CCN(Cc3ncccc3C(=O)O)C2)=O)cc(F)c(F)cc1F Cc1c(N)ccc(C(N2CCCCC(N(C)C(c3cc(O)nn3C)=O)C2)=O)c1F CCCC(CC)C(=O)NC(C)(C)CNC(c1cnn(Cc2ccccc2Cl)c1)=O C1(COC)CCN(C(c2cncc(CNC(=O)Cc3csc(C)c3)c2)=O)CC1 c1(C(N(CCOC)CCNC(=O)C(C)NS(=O)(=O)CC)=O)cccn2nccc12 C#CCCCC(C)C(=O)NC(C(=O)NCC(CC)CC)C1CCCO1 C(=O)(CS(=O)(=O)N1CCN(C)CC1)N(CC(CC)NC(CSCC)=O)C N1(C(C(C2CCOC2)OC)=O)CCC(C)N(C(=O)CCCN2CCCCC2)CC1 c1(C(=O)NCCN(C(C(C=CC)O)=O)CC(C)O)ccc(CCC(N)=O)cc1 C12(C(N(CC#C)CCF)=O)CCC(CC1)N(C(c1ccc(Cl)cc1)=O)C2 N1(C(CCCCCCSC)=O)CCC2(CCC(NC(C3CCSC(C)C3)=O)C2)C1 c1(NC(CCN(C(CCC)C)C2CC2)=O)ccc(CN(CC)CC2CC2)o1 N1(C(C)=O)CCOC(C(=O)NC(c2cccnc2)C)C1 CC1(C)COCC(C(=O)NC2CN(C(C3(C)CC(C(F)(F)F)C3)=O)C2)O1 c1(C(=O)NCCCCC2CCN(C(c3n(C)ccn3)=O)CC2)ccc(F)cc1Cl c1(OC)cc(C(C(=O)NCCN2CC[SH](F)C2)N(C)C)ccc1C#N N1(C(c2ccn(CCCC)n2)=O)CCN(C(c2cc(Cl)cnc2O)=O)C(C)C1C c1(CC)nc(C)ncc1C(=O)NC(C)CC1CN(C(c2nccnc2C)=O)C1 C1(CNC(C2N=C(C)SC2)=O)CN(C(=O)C(n2nc(C)cc2C)C)CCCO1 c1(OC)cc2c(cc1C(=O)NC(C)C(CO)NC(c1cc(C#N)on1)=O)OCO2 N1(C(CN(C)CC)=O)CC2CC(NC(=O)CCC3CCCCN3C)C(C2)C1 c1(OC)ccnc(C(=O)NCC(C)(C(C)C)NC(C2CC(O)CN2C)=O)c1 c1(C(=O)NC(C2CCN(C(Cc3c(C)nc[nH]3)=O)CC2)C)cc(Cl)nnc1Cl N1(C(c2ccc(OCC)nc2)=O)CCCC2(CNC(=O)CN(C)C(C)=O)CC12 N1(C(C2CCC(C)CC2)=O)CCCCC(NC(=O)C=Cc2cc(C(N)=O)co2)C1 c1(CN=c2ccnc(NCCC3CCC(C)CC3)[nH]2)c[nH]c2ccc(F)cc12 n1(CCOC)nc(C(=O)NCC2C(C)CCN2C(=O)CCS(C)(=O)=O)ccc1=O Cc1cccc(C(=O)Nc2cccc(NC(C3CCCC4CC34)=O)c2)c1Br c1(N2CCC(N(C)C3CC3)C2)nc2c(c(=NCCc3cn[nH]c3)[nH]1)SCC2 N1(C(c2cc(C)[nH]n2)=O)CC2(NC(=O)CC(C)c3ccncc3)CCC1CC2 C1(OCCNC(=O)NCC(C2CCCCO2)(C)C)CCCOC1 N1(C(C(C)(F)F)=O)CC2CCN(c3ncc(I)cn3)C2C1 C1(S(=O)(=O)c2ccccc2)(CNC(=NC)NCC2C3CCC(C3)C2(C)C)CCCC1 CCC(C)(COC)C(=O)NCCC1CCC(NC(C2(CN(C)C)CC2)=O)C1 c1(C(C(=O)NC(C)CNC(c2c[nH]nc2C(F)(F)F)=O)(F)F)ccc(Cl)nc1 N1(C(=O)Nc2cc(C(=O)OC)cc(C3CC3)c2)CCCC(C2CCCCC2)C1 C1(CCNC(C2C(CCOC)C2)=O)CN(C(=O)C(N2CCCCC2)C)CCO1 c1(CC)cccc(C(=O)NC(CN(C)C(c2ccc(CN(C)C)[nH]2)=O)CC)c1N C1(C)(CNC(C(CCC)N(C)C)=O)CCCN(C(c2cnc(C3CC3)[nH]2)=O)C1 CCC(CC)CC(F)C(=O)NC1COCC1NC(=O)C(=Cc1ccncc1)C C1(NC(c2c(C)oc(CO)c2)=O)(CNC(=O)CC(=O)NC2CC2)CCCCC1C CCC(F)(F)C(=O)NCC1C2CN(C(=O)C(C)(C)CC)CC12 C(=O)(CC(C)C(F)F)NCCN(C(=O)CC1CCC(C)CO1)CC C1(NC(C2CC(C(=O)OC)C2)=O)CCN(CCNC(=O)C(C)=C2CCCC2)CC1 N1(C(c2n(CC#C)ccc2)=O)CCC(C)(CC(=O)NC2CCC(F)(F)C2)C1 C1(CSC)CCC(C(=O)NC2(C(N3CCCC3CN=[N+]=[N-])=O)CC2(C)C)CC1 CCCC(C(O)C(=O)N1CCC12CCC2)NC(=O)C(C)(CO)OC N1(C(c2cn(CC)nc2)=O)CCC(N=c2nc[nH]s2)C(CC)C1 N1(C(COCCCOC)=O)CCC(CNC(c2cnnc(O)c2)=O)C12CCC2 C#Cc1cc(C(=O)NCc2ccc(CS(N)(=O)=O)cc2)ccc1C C(=O)(C1Cc2ccc(Cl)cc21)NCC1CCC(CNC(CC(C=C)(C)C)=O)CC1 c1(C(=O)NCOC(=O)CN2CCCC(NC(c3ccoc3)=O)C2)ccccc1C#N C1(C(=O)NC(C2(CNC(=O)CCC(=O)N3CCOCC3)CC2)C)CCSC(C)C1 N1(C(=O)CNc2ccccn2)CCOCC1C1CCN(C(=O)C(O)C2CC2)CC1 C=C(CNC(=O)Cc1ccon1)CCNC(=O)OC(C)(C)C.C1CCC(=O)N1 c1(C(=O)NCC(C)N(C)C(c2ccc(F)c(C(F)F)n2)=O)cc2n(c1)CCCC2 Cc1cnc(C(N2CCC(C)(C)C2C(=O)NOCC2CC2)=O)c(F)c1 c1(CC(N2C(CC)CN(Cc3cccnc3C)CC2)=O)[nH]nc2c(Cl)cccc12 Cc1cc(C)c(C(=O)NC2CC3(C2)CN(C(C2(C)CCSCC2)=O)C3)c(C)n1 C(=O)(CC(C(F)F)C(C)(C)C)NC1C2N(CC1)C(=O)CS2.c1(CC)cccs1 C(C)(C)(C(C)CC(=O)NCc1cc(Cl)ccn1)NC(c1n(CC#C)cnn1)=O Cn1nc(C(N2CCCNC(=O)C2)=O)c2c(-c3ccc(F)s3)cccc12 N1(CC(COc2cccc(N(C)C)c2)O)CCSCC(CO)C1 CC(C)CC(CNC(C1CN(C(C2CC2C(F)(F)F)=O)C1)=O)NC(N)=O C1(NC(c2c(SCC)cncc2)=O)CCN(C(c2ccn(C)c2C)=O)CC1CO Cc1nc[nH]c(=NCC2(C)CCN(C(C3(C)CCOC3)=O)CC2)c1F c1(CCC)[nH]nc(C(=O)NC2CCC2NC(=O)CCC2CC2(C)C)c1[N+](=O)[O-] N1(C(CCS(C)=O)=O)CC2CN(C(=O)C(C)(C)Cc3cnn[nH]3)CC2C1 C1(NC(CC(COC)NC(=O)C(C)(F)c2ccon2)=O)CCCCC1N=[N+]=[N-] CC1(C(=O)NCC2(F)CN(c3nnc(C(F)(F)F)s3)C2)CCNC1=O Cc1cccc(C)c1CC(=O)NC1COCC1NC(=O)COc1ccccc1 O=S(=O)(c1c[nH]ccc1=NC1=CCCSC1)NC(CC1CCCCO1)CO C(=O)(C1=C(C)OCCS1)N1CCCC(N(C(C2(C)CCC2C(=O)OC)=O)CC)C1 c1(C(N2CCC(c3nc(-c4ccncc4)no3)CC2)=O)ccc(C(F)(F)F)nc1Cl c1(C(c2nnnn2CCCC)NCC(CC(=C)Br)(C)C)cc(C#N)ccc1F C(=O)(CCS(=O)(=O)N(C)C)NCC(N(C(CNc1c(C)cncc1)=O)C)C1CC1 C(CCCCCC(=O)NC(C(=O)NC(C)C)C(C)C)NC(C(CC)COC)=O C(C#Cc1cn(CC2CCCOC2)nn1)NC(CCc1nnc(C)n1C)=O n1(CC(=O)NCC2(F)CN(C(C3CCC=CO3)=O)C2)nnc(C2CCCC2)n1 C1CCC(C)C(=O)O1.C1(CO)(CO)CNC(=O)C2CC(OC)CN12.C(C)(=O)OC Cc1[nH]c2ccccc2c1CN1CCC(CN2CCS(=O)CC2)C1 c1(N2CCC(NC(c3c(CC)[nH]cc3)=O)(CF)C2)cc(Cl)nc(C)n1 c1(CC(N2C(CNC(c3cnn(C4CC4)c3)=O)CCC2)=O)ccc(O)nc1.N1CC1 N1(C(C2C(C)(C)C2)=O)CCC(CNC(=O)CC2(O)CCC2)C12CCC2 N1(C(C(C)NC(=O)C(O)CC(C)(C)C)=O)CCC(CO)C(C)(C)C1 C1(CNC(Cn2cc(C(C)=O)nn2)=O)CC(O)CN1C(C1CCCCC1)=O c1(C(=O)NC2(CCNC(C=CC=C)=O)CC2)cnn(Cc2ccccc2)c1C1CC1 C1(C(N(C)CC2(O)CCN(C(CC3CC(SC)C3)=O)C2)=O)CN(CP(C)(C)=O)C1 C1(NC(CC(C)O)=O)CN(C(c2ccc3cnoc3c2)=O)C2(CCCCC2)C1 C1(NC(c2c(C)cccc2Cl)=O)CN(c2nccn3nnnc23)CC2(CC2)C1 Cc1cc(O)ncc1C(=O)NCCN(C(=O)COc1cn[nH]c1)CCOCCO c1(C(=O)NCC2CC(NC(c3cccc(NCC)c3)=O)C2)n[nH]c2c1COC2 C=CC1(C(N2CC(OCCNC(C3C4C5CCC(C5)C34)=O)C2)=O)CCCCC1 C1(NC(C(CC)=CCCC)=O)CCN(C(c2ccc(C3CC3)cc2F)=O)CC1O c1(N(C2CC3CNC2C3)C(c2ccc(C)s2)=O)cccc(C)c1F C(C(=O)NCCn1ccnn1)(C1=NOCC1)N1CCC(C(=O)NC2CC2)C1 C1(NC(C2C(C#N)C2)=O)C2CC3CN(C(c4ccc(OC(F)F)cn4)=O)C1C3C2 CC(F)(F)C(C)(C)CC(=O)NCC12CCC(CC1)CN2C(=O)Cc1nc[nH]n1 C1(CNC(C2OCCN(CC)C2)=O)CN(C(c2cnc(C(F)F)s2)=O)CC1(C)C N=c1[nH]nc(CCC(N2CC(CO)(NC(=O)CN3CCCCCC3)C2)=O)s1 Cc1cnc(C(C(=O)NC2COC2)N(C)CCc2ccccn2)s1 C1(C)(NC(CC2C(C)C2)=O)CCN(C(C2CC(OC3CC3)C2)=O)C1 C(=O)(C(F)(F)C(F)F)NCC1N(C(c2cc(C3CC3)on2)=O)CC1 c1(C(=O)NCCCCNC(c2c[nH]c(=N)o2)=O)cn(CC#N)c2ccccc12 C1(C(N2CCC(CCC(=O)N(CC(COC)O)C)C2)=O)(OC)CCCCC1 N1CCCCC1C1CCN(CC2(O)CCCOC2)C1.Cn1cccc1C=O C1(C(=O)NCC(CNC(C2CC2(F)F)=O)C(F)(F)F)CCC2(CC1)CC(O)C2 N1(C(CCN(C)CCO)=O)CC(NC(C2CCCNS2(=O)=O)=O)C(C)(C)C1 C(C(C)(C)CC(=O)N1CCC(c2ccon2)C1)NC(C1C(OC)(OC)CC1)=O C=C(Cl)CCC(=O)N(C1CCC(NC(c2cccc(-n3cc(C)cn3)c2)=O)C1)C N1(C(CC(C=C)(C)O)=O)CC(C(=O)Nc2ccc(F)c(C(N)=O)c2)CC(C)(C)C1 C(c1ccncc1)=CC(=O)N(C)CC1CCN(C(C23CC(Br)(C2)C3)=O)C1 C1(NC(C(C2CCCOC2)OC)=O)CC(O)C1CC(=O)N(C)C c1(C(=O)OC(C)(C)C)cccc(NC2(c3cccs3)CC2C)c1 CC1CC(O)CCN(C(C2CCC(O)CN2C(=O)COCC(F)F)=O)C1 c1(C(=O)NC23C(CN(C(C(C)C4(O)CCC4)=O)C2)C3)ccc2cnsc2c1 N1(C(C=CC(c2ccc(C)cc2)=O)=O)CC2OCC(NC(=O)C3=C(Cl)CC3)C2C1 C1(C(=O)NCCOCCCNC(=O)COc2ccsn2)COCCOC1 C1(CNC(CNC(CNC(C)=O)=O)=O)CCCN(C(=O)CC2C=C2C)C1 Cc1ccn2cc(Nc3cc(NCCC4CCCO4)nc(C)n3)nc2c1 C(=O)(C(C(C)(C)C)c1ccc(F)c(C)c1)NCCNC(C1(CC=C)CCCC1)=O N1(C(C(C)C(C)(C)C)=O)CCC(F)(F)C(CNC(=O)CCCc2cc[nH]n2)C1 C1(CNC(c2cnc[nH]2)=O)CCN(C(=O)Cc2cc(Cl)cc(Cl)c2)C12CC2 Cc1ccc(Br)c(-c2nnc(NCCN3C(C)CCCC3C)o2)c1 CC(=O)CCC(=O)N1CCC(F)(CNC(c2ccccc2-n2nccn2)=O)C1 C(=O)(C1=CCCCC1)NC1C(NC(=O)CCCN2CCCC2)COC1 C(C(C)(O)CNC(C1CCC1NC(c1cnsc1C)=O)=O)SC C1(C(=O)OC(C)(C)C)CCN(C(=O)C(=O)NC2CC3CC4C(C3)C24)CCO1 N1(C(c2c(CC)nns2)=O)CCSCC1CCNC(=O)Cc1ccsn1 Cc1nc(N2CCC(C)C(NC(c3ccc(CF)cc3)=O)C2)ccc1C#N c1(CCC(=O)NC(C2CCN(C(c3cncc(O)c3)=O)CC2)C)ccc(O)cc1 N1(C(c2cc(C)n(C3CC3)n2)=O)CCC(C)N(C(=O)CC(O)C(C)(C)C)CC1 Cc1ccc(C(=O)NC2CCC(CC(=O)N(CCF)C3CC3)C2)cc1C#N C1(CC)(NC(=O)CN2CC(=O)N(C)C2=O)CCCN(C(C2CC2C(C)O)=O)C1 c1(C(=O)NC2C(NC(CCN(CCCCC)C(C)C)=O)C2)nc(C2CC2)oc1C.OCC C(=O)(CC(C)(C)C#N)N1CCCC(CCC(=O)N(CCC#N)C)C1 c1(OCC(=O)NCC2N(C(C3(C=C)CCOCC3)=O)CC2)cc(C)c(Cl)c(C)c1 c1(CCCN(C)C(=O)NONC(=O)OC)cc(OC)cc(Cl)c1F C1(C(=O)NCc2cccnn2)CC12CCN(C(=O)CC1COCCO1)CC2 CCC(CC)(CCNc1ncc(C)cn1)NC(C1CC2C=CC1CC2)=O N1(C(Cc2c(C)scc2)=O)CCCC(CNC(=O)Cc2cncc(F)c2)C1 N1(C(=O)NCC(c2cccc(Cl)c2)(F)F)CCCC(C2COC2)C1 C(C(=O)NNc1ccccc1SC)(c1ccccc1)N(C(c1cnn(C)c1)C)C N1(C(CCC2(C)CCCN2C(=O)Cc2cnn(CCF)c2)=O)CCc2ccsc2C1 C(C1(C)CCCc2ccccc21)NC(C=Cc1c(C)n(C)nc1)=O c1(OCOC)cc(-c2cnc(CC(=O)Nc3ncncc3Cl)nc2)ccc1C N1(C(C2C(CCOC)C2)=O)CC(CNC(=O)C=CC2CCCCC2)CCC1C C(=O)(CC(CNC(=O)C(C)C#N)OC)N(CC#C)C(C)C N1(C(C2(OC)CCS(=O)(=O)C2)=O)CCC(C)C(C(=O)NCc2cc(Cl)ncc2F)C1 C1(C2CCOCC2)(C(N2CCC(N3CCN(c4nnco4)CC3)CC2)=O)CC1 N1(C(CC(C=C)CC)=O)CCC2(CCC2)C(NC(c2ccc(C)nn2)=O)C1 C1(NC(CN(C(C(C)=C(CC)C)=O)C(C)C)=O)CCOCC1C c1(N2CCC(NC(Cc3ccc(C(CC)=O)cc3)=O)C2)ncc(C(C)C)cc1C#N c1(C(C(=O)NC(C)(C)CC)N(C(C)C(=O)OC)CC)ncc(C)cc1C c1(CC)nc(C)c(C(=O)N(CCC(C)(C)NC(c2cnc(C(C)C)[nH]2)=O)C)o1 c1(-c2n(CC3N(C(C4CCC(F)C4)=O)CCC3)ccn2)c(F)cccc1Br c1(CC)cccc(CC)c1C(=O)NC1CN(C(=O)CCC2CCCOC2)CC1C C(=O)(CC(C)(C)c1cccs1)NC1(C2N(C(Cn3c(C)nnn3)=O)CC2)CC1 c1(C(=O)NCC(CC)NC(=O)CC2CCC(CC)O2)cc(Br)c(F)cc1Cl c1(C(N2CCC(CO)(OCC)C2)C(=O)NCC)ccc(C(F)F)c(Cl)c1 c1(NC(C2(SC)CC2)=O)cccc(C(C)=O)c1.C12(CCCC1)C(=O)NC2 c1(CNC(C2CCN2C2CC2)=O)cc(O)cc(O)c1 C(CCN=C(NCC1OCC1(C)C)N1CCC(CC(F)(F)F)C1)OC(C)C c1(NC(C2(C)CCN(Cc3ccc(C#N)cc3Cl)C2)=O)nc(Cl)c(Cl)cc1Cl c1(C(N2CC3C(CNC(C(=C(C)C4CC4)F)=O)C3C2)=O)coc2ccc(F)cc12 N1(C(CNC(Cn2ncc(CC)c2)=O)C)CC(O)CC1C N1(C(c2ccc(O)nc2)C(=O)NCCC(=O)OCC)CCC(O)(CC)CC1 c1(C(N2CC=CC(NC(CCCNC(N)=O)=O)C2)=O)cc(F)c(F)cc1O N1(C(CC#N)=O)CCCCC1C1CCCN1C(C1CC2(CCCC2)C1)=O c1(C(N(CC(C)NC(=O)CSCc2ccc(Cl)cc2)C)=O)c(N)sc2c1CCC2 N1(C(CCC(=C)Cl)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCC(C)OCC)C1 CC(C)(CNC(c1cc(Cl)c[nH]1)=O)CC1CN(C(C2CCCO2)=O)C1 C1(NC(c2c(C)onc2CO)=O)COC2(C1)CN(C(=O)CC1(C)CC1)C2 Cc1cnc(C(=O)N(CCNC(=O)CCc2scnc2C)C(C)C)c(Br)c1 c1(C(=O)NCc2c(OC)c(C)ccc2)cc2n[nH]cc2cc1-c1cnoc1 N1(C(COc2c(C)ccc(C)c2)=O)CCCC12CCN(C(=O)C(C)(O)C1CC1)C2 CCC(C)C(C)(O)CNC(=O)NC1C2CN(c3ccccc3)CC12 C(CCCCC(=O)NCC1CC(F)(CNC(C2CCCC2C)=O)C1)SC c1(C(=O)NCCC2CCN(C(c3c(O)cccc3Cl)=O)C2)cccc2occc12 C(=O)(CCNC(=O)C(C1(C)CC1)OCC(C)NC(=O)OC)OCC CC(C)CC(C(=O)NC1CCC(SCc2cnn(C(C)C)c2)O1)ON.S(C)(=O)(=O)N CC(CNC(=O)CCc1csnn1)C(=O)N(CC(=O)NC1CC1)C C1(NC(CC(C)n2cccn2)=O)CN(C(c2cnns2)=O)CC2(CC2)C1 C1(C)(CNC(CCC2(C)CN(C(=O)CC#N)C2)=O)NC(=O)NC1=O C(C)(C)(CC(=O)N1CCCC1CN(C(=O)C(F)CC1CC1)C)N(C)C N1(C(C(C)OC)=O)CC2(CC(NC(=O)C(F)OC(F)(F)F)C2)C1 N1(C(C(C(CC)C)N)=O)CCn2c(nc(C(=O)NCC3CCCN(C)C3)c2Cl)C1 N1(C(C(C(C)O)N(C)C)=O)CC2=C(C1)CN(C(=O)CCc1ccc(N)c(N)c1)C2 N1(C(c2cc(C(F)(F)F)nn2C)C(=O)NCCOC)Cc2ccnn2CC1C C1(C(CC)C)CCCN1C(=O)CC.c1(N)cncnc1.C1(=O)CSCCN1 Cc1cc2nc(NC(N3CCC(C(C)(C)C)CC3C3CC3)=O)[nH]c2cc1Br Cc1cc(F)ccc1C(=O)NC1(C)CCCN(C(C2(C(F)(F)F)CC(O)C2)=O)C1 CC1OCCC1CC(N1CC(O)(C(F)C(=O)N(C2(C)CC2)C)C1)=O C(=O)(C1=NOC2COCC12)NCC(CC=C)NC(c1cn(C2CC2)nn1)=O C(=O)(C(C)(C)CS(N)(=O)=O)NC(C(CO)NC(c1n(CC)c(O)nc1)=O)C C1(C(=O)Nc2ccc(F)nc2)CCCC12CCN(Cc1cc(Cl)cc(Cl)c1Cl)C2 c1(C(N(C(CNC(C(CSC)OC)=O)C)C)=O)c(-n2cccn2)cccc1F c1(C(N2CC(C(C)NC(=O)CNC=O)OCC2)=O)c(F)cc(F)c(F)c1F C1(NC(c2cccc(COC)c2)=O)CCN(C(C2(CC3CC3)CCC2)=O)CC1F O=S(=O)(c1cccnc1N1CCC(F)(CO)CC1)NC1CC2(C1)CC21CCC1 C(=O)(N=c1ccc(I)n[nH]1)N(C(C(CCC)C)C)C c1(C(=O)OC)ccc(CN2CC3(CN(C(C4(C)CCOCC4)=O)C3)C2)c(Br)c1 c1(C(N2C(C)CC(NC(=O)CCS(N)(=O)=O)CC2)=O)nc2ncccn2n1 CC1C(NC(=O)Cc2ccnc(F)c2)C(C)CCN1C(c1ccc(C#N)cc1)=O N1(C(C=CCN(C)CC)=O)CCCC12CN(C(=O)C(C1CC(F)(F)C1)O)C2 CC(C)(C(=O)NCC1CCCC1NC(C1CC1(Cl)Cl)=O)C(N)=O CCCCCC(O)C(=O)N1CCC2C(C1)CN2C(=O)CP(C)(C)=O N1(CCC)CCC(C(=O)NCc2n[nH]c(=N)s2)(OC)CC1 c1(C(=O)NCCNC(c2cc3ncccc3o2)=O)snc2ccccc12 c1(CNC(=N)NCCc2cn[nH]c2)cc(Cl)c(Cl)cc1Cl c1(C(N(CCCCCCNC(C2CCOC2=O)=O)C)=O)ccc2c(c1)CCO2 CC1CN(C(C2CCC(CNC(C3CCNC(=O)C3)=O)CC2)=O)CC(C)(C)O1 c1(C(=O)NC(C2(C(=O)NCCCCOC)CC2)C)cc(O)cc(F)c1 c1(OC)ccc(OC)c(C(O)C(=O)NCCN(C(=O)CC(C)C)C(C)C)c1 Cc1ccc(CC(=O)NC2CC(CC(=O)Nc3ncco3)C2)o1 C(CCCCCC(=O)N1CC(NC(C2CN(C)CCO2)=O)C(SC)C1)SC N1(C(c2nc(C(C)C)sc2)=O)CC2C(CCCC2NC(=O)C(C)c2ccco2)C1 Cn1ccc2cc(S(=O)(=O)NCCCCCc3ccccc3)ccc12 C(=O)(C(C)(C)C(=O)NCC)N(CC(C(=O)N(C)Cc1onc(CC)n1)C)C c1(OC)ccc(C(C)C(N2CCC(NC(C3CC=CCO3)=O)CC2)=O)cc1OC c1(OCC(N2CC3(C(NC(C4CCC4)=O)CCC3)C2)=O)ccc2ccccc2c1 Cc1ccccc1-n1nc(-c2ccc(F)cc2)nc1-c1cn(C)c(O)n1 C1C(C(N(CC(C2CCCC2)O)C)=O)CC(c2ccccc2)S1 N1(C(CN(CCC)C(c2nccs2)=O)=O)CC2CCC(O)C2C1 CC1COCCC1N(C)C(=O)OC(C)(C)C.c12cnc(s1)CN2 c1(C(=O)NC(CNC(C2(CC=C)CCCC2)=O)(C)C)scc(C)c1OC N1(C(C2(CC=C)CCN(C(=O)CC3CSC3)C2)=O)CCC(C(=O)NC)CC1C O=C(C1=COCCC1)NCC(O)CNC(c1cscc1C(F)F)=O N1(C(CC(C(=C)C)OCC)=O)CC2(CCCC2NC(C2CCC(N=[N+]=[N-])C2)=O)C1 C1(NC(c2cc(CC)no2)=O)CCC(C)N(C(=O)Cc2csnc2C)C1 C1(CSC)CCCN1C(C1CCC(NC(=O)C=C(C)C2CC2)C1)=O Cc1ccc(OCCC(=O)NCCN(C(C2CC=C2C)=O)C2CC2)cc1C N1(C(CCC(=C)Br)=O)C2CCC1CN(C(=O)C(C)Oc1ccc(F)cc1)C2 C1(C(=O)NCC2N(C(CC(C)c3cccnc3)=O)CC2)CC(=O)OC1(C)C C1(C)(CNC(c2c(OC)csc2)=O)CCN(C(C2(c3ccccc3Cl)CC2)=O)C1 Cc1cccc(CCC(=O)NC2CCC2CNC(=O)CC(C)(C)C)c1Cl c1(C(N(C2CCCN(C(Cc3c(C)n[nH]c3)=O)CC2)C)=O)cc(F)cc(F)c1N c1(C(CC(=O)NC2CC(CNC(CCOC)=O)OCC2)O)cc(Cl)cc(Cl)c1 C1(C(=O)NCC(CNC(C2(C#N)CCC2)=O)CO)CC2CCCCCC12 n1(CC)nc(Br)nc1C(N1CCOC(CC)C1)C(=O)NCC1C(F)(F)C12CC2 N1(C(c2c(CC)n(C)cc2)=O)CCC(CNC(=O)C(O)C(C)(C)C)C(O)C1 C1(NC(C2CC23CC(O)C3)=O)CCCCN(C(c2c[nH]nc2C(F)(F)F)=O)C1 c1(C(N2CCCC(N(C(C(C)OCC#C)=O)C)C2)=O)ccc(F)cc1C c1(C(C)=O)ccc(C(=O)N(CC(=O)Nc2cnn(CCF)c2)CC#N)cn1 C(=O)(C(CC)CCOC)NCc1ccc(C(N(C(CC)CC)C)=O)s1 N1(C(C2(C#C)CCC2)=O)CC2CN(C(c3cc(F)ccc3CC)=O)CC2C1 c1(C(=O)NC2C(C)CN(C(C3CCCC3O)=O)C2)cccc2nc[nH]c12 c1(C(N2C(CNC(CCc3cccc(C)c3)=O)CC2)=O)csc([N+](=O)[O-])c1 C12(CNC(c3c(N)cccn3)=O)CCCC1CN(C(=O)CCc1cccs1)C2 N1(C(c2cc(CC)c(F)cc2)C(=O)NCC(C)C)CCC2(CCCCN2C)C1 C1(C(N2CCC(CCN3CCCCC3CCO)C2)=O)CCC12CCCO2 c1(OC)cc(C(C)NC(C)C(=O)Nc2cccc(SC)c2)cc(OC)c1O c1(C(N(CCCN(C(CN(CC)CC)=O)C)C)=O)csc(C)c1C1CC1 Cc1ccc(CC(C(=O)NC2CCC(F)(CNC(=O)CC3CC3)C2)C2CC2)cc1 n1(CC)cccc1C(=O)NCCCCNC(C1(C)C=CCC1)=O C(=O)(C(O)C(C)(C)C)NC(C)CCCCNC(C1NC(=O)OC1C)=O C1(F)(C(N(C)CCOCC2CC2)=O)CCCN(C(C2(C(F)F)CCCO2)=O)C1 c1(C(N2CC(C)(CNC(C(CCN(C)C)O)=O)OCC2)=O)c(F)ccc(F)c1F C1(CNC(C(Cc2ccccc2)OC)=O)CC(SC)CN1C(=O)C(C)C CCCC(CC)CCC(=O)N1CC(F)(CNC(=O)C(C2CCC2)OCC)C1 Cc1nn(C)cc1C(=O)NC(C)(C)CCCNC(=O)CC1CC1(C)C c1(CC)cc(C(N2CC(OC)C(NC(C3CC(=C4CCC4)C3)=O)C2)=O)ccc1N C(=O)(CCCCC(C)C)NCC1C(CC)CCN1C(=O)CC(=O)NC(C)(C)C S(=O)(=O)(c1ccc(NC(=O)C(F)(F)F)cc1)N1CC(C)OC(C(N)=O)C1 N1(C(COCC(C)C)=O)CCc2ccc(CNC(C3CCC(C)C3)=O)cc2CC1 c1(CN(C2CCCC2(F)F)C)ccc([N+](=O)[O-])cc1C CC1CCC(NC(C23CC(C(F)F)(C2)C3)=O)CN1C(=O)CCn1cnnn1 C(=O)(CC(C)C(F)(F)F)N1CCCN(C(c2ccc(C(=O)OCC)nn2)=O)CC1 c1(CC(N2CC(CNC(=O)C(C3CC3)C3CC3)OCC2)=O)csc2nccn12 N1(C(C(C2CCCCC2)NC(=O)C(c2ccccc2)F)=O)CCc2ccncc2C1 C1(OC)CC(CNC(=O)C=Cc2cc(C)no2)N(C(=O)CC2(O)CCOC2)C1 N1(C(c2cccc(SC)c2)=O)CC2CCC1CN2C(C1CC(C)=NO1)=O c1(OC)ccnc(F)c1C(=O)N(CC(C)NC(=O)CCC(C)C)C c12ccc(c(F)c1)NC21CC1.C(=O)(CC(C)N(C)C)OC C(C)(CO)(CN=c1ccc(S(=O)(=O)N(C)C(c2ccco2)C)c[nH]1)OC n1(CC)nc(C(N2CCC(NC(c3sccc3OC)=O)C2)=O)cc1O N1(C(c2c(C)nsc2C)=O)CC2CN(C(c3ccnn3C(F)F)=O)CC2(C)C1 N1(C(CCC(=O)OCC)=O)CC2(NC(C3CCC(C)(C)O3)=O)CCC1CC2 N1(C(c2ccc(O)cn2)=O)CCC2C(C1)CN2C(=O)Cc1csc2ccccc12 CCC(CC(=O)NC1C=CC(CNC(c2cc(C)sn2)=O)C1)CC(C)C c1(COC)nc(NC2CCCSCC2)cc(=NCC2CCCC2(F)F)[nH]1 N1(C(C(CC#C)O)=O)CC2CC(C1)CN(C(C1COCCN1CC)=O)C2 C1(NC(C2(C)CCC2)=O)CC(F)CN(C(=O)CC2(c3ccccc3)CC2)C1 C#Cc1cc2c(cc1C(=O)OCc1nc(C(=O)OC)co1)OCO2 N1(C(CCNC(COC)=O)=O)CC(CNC(c2csc(C)c2C)=O)C(O)C1 c1(C(N2C(C)(CNC(C3(OC)CC3)=O)CCC2)=O)ccc(C)c(F)c1N C(=O)(CC(C(F)F)NC(=O)C(C)=C1CCC1)N1CC(CCC)OCC1 C(C(C)(C)CC(=O)NCC1CC(NC(=O)CSCC(N)=O)C1(C)C)OC N1(C(CC2CC(=O)NC2)=O)CC2C(C(F)(F)F)CC2(NC(c2cnccn2)=O)C1 O(N=C(N)c1ccc(F)cc1)CC1(NC(CNC(C(C)(C)C)=O)=O)CC1.C1CO1 c1(CC(=O)NC(C(=O)N(C(c2ncc(C)o2)C)C(C)C)C)cccc(O)c1 C1(COC)(COC)CCCN1C(c1ccc(C(=O)CCC(C)NC(C)=O)o1)=O c1(CC)[nH]nc(C(N2CCOC(CCNC(=O)CN3C(C)CCC3C)C2)=O)c1C CCC(CC)CC(F)C(=O)NC1CCC1CNC(C1COC(C(C)C)C1)=O C1(C(N(C2CCCC2)C)=O)C2CN(C(C3CC(C)(C)CO3)=O)CC12 C1(C(=O)NCC(C)(C2CC2)NC(c2ccncn2)=O)CCCS1(=O)=O c1(C(Cc2cncnc2)CNC(N2CCC(CB(O)O)C2)=O)ccc(Br)cc1 Cc1ccnc(F)c1NC(C1CC1C(=O)Nc1c(Cl)ccnc1Cl)=O C1(N(C(=O)C=Cc2ccoc2)C)CC2CCC(C1)N2C(C1(C)CCOC1)=O C1(O)(CC)CN(C(=O)C(O)CNC(=O)CSCC(F)(F)F)C1 Cc1cc([N+](=O)[O-])ncc1C(N1CCSCC1CCNC(=O)Cc1cc[nH]n1)=O C1(C(=O)NCCC(C)NC(c2c(CCC)nns2)=O)COCC(C)(C)O1 c1(CCC(N2CCC(Cn3cc(C(C)(C)OC)nn3)C2)=O)ccc(Br)cc1F C1(C(N2CCN(C(CC)=O)CC2)=O)CC(C)(C)CN1C(=O)CC(C)CN(C)C c1(C(=O)NCCNC(=O)CN2CCCC2=O)ccc(SC2(COCC)CC2)cc1 c1(N2CC(C)CN(C)CC2)nc2c(c(=NC3CC(F)(F)C3)[nH]1)CCC(C)CC2 CCC(C)(CNC(=O)C(C)C(F)F)C(=O)N1CC(n2ccnn2)C1 N1(C(=O)CCc2cnccn2)CC2(CCCN(C(C34CCCCC3C4)=O)C2)C1 c1(C(=O)NC2CN(C(c3cnc[nH]3)=O)CC23CC3)c(F)cc(Br)cc1Cl N1(c2c(C)cnc(C)n2)CCC2C(CCCN2C(C2(n3ccnn3)CC2)=O)C1 C1(OCC#C)(NC(c2cnn(CCNC(=O)NCC=C)c2)=O)CCOCC1 c1(C(=O)NCCC2(CNC(c3csc(C4CC4)n3)=O)CC2)nc(C2CC2)cs1 c1(C(=O)NCC2N(C)CCN(C(CCN(C)CC)=O)C2)ccc2[nH]nc(O)c2c1 N1(C(C(N2CCCNC2=O)C)=O)CC=C(CNC(C2CCCCCN2C)=O)CC1 [N-]=[N+]=Nc1ccc(-c2cn(CCC(N3C4CCC3CC(O)C4)=O)nn2)cc1 N1(C(CCCCC#C)=O)CCC2CN(C(=O)C(CC)CC(C)C)CCC12 C1(CC)CN(CC)CCN1C(c1csc(CNC(=O)C(C)c2ccco2)n1)=O C1(NC(Cn2c(C)ccn2)=O)CCN(C(=O)CCCC(=O)NC(C)C)CC12CC2 C12(C(=O)NCCN(C(=O)Cc3csc4nccn34)CCOC)CC(C1)S(=O)(=O)C2 N1(C(c2nc(C)cnc2C)C(=O)NCCSCC)CCC(C)C2(CCCCC2)C1 Cc1nc(CO)sc1C(N1CC(CNC(C2(CF)CC(F)(F)C2)=O)C(C)C1)=O C(=O)(C1=CCCS1)NCC1C(CNC(C2(CO)CCOCC2)=O)CCCC1 C(=O)(C(C(=O)OCCN)C(C)(C)C)NCC(N(C(=O)COc1ccsc1)C)C1CC1 c1(OC)cc(F)c(I)cc1C(=O)NCc1ccc(Cl)c(Cl)c1C C1(NC(c2c(OC)cc(O)cc2)=O)CCN(Cc2ccc(OC)cc2)CC1(C)C C1(NC(C2CCS(=O)(=O)N2)=O)CCCCC12CCN(c1nc(C3CC3)ns1)CC2 N1(C(c2nncc(OC)c2)=O)CC2(CC2)CC1CNC(C1(CO)CCC1)=O C(C)(C)(CCCCC(=O)NC(C)(C)C)NC(C(COC)C)=O c1(NC(c2nnnn2C2(C)CC2)(C2CCCO2)C)ccc(N)cc1F.C(CF)OCC c1(SCC(N2CC(NC(c3cc(OC)ncc3)=O)C2)=O)nn(C)c(=O)n(C)c1=O Cc1nn(C2CC2)cc1C(=O)NCCCNC(C1(C(C)(C)O)CCC1)=O N1(C(=O)Nc2ccc(C)cc2)CC2CN(C(=O)CN3CCCC3=O)CC12 N1(C(CCC=CC)=O)CCC(NC(=O)Cc2ncc(C)[nH]2)C2(CCC2)C1 C(C)(C)(CC(=O)N1CCC(Oc2ccccc2)CC1)n1cc(CC(CC)C)nn1 c1(C(=O)NC(C)CN(C(=O)C(C)(C)N(S(C)(=O)=O)C)C)nc2c(s1)COCC2 c1(N(C)C)cnc(C(=O)NCC2(O)CN(C(C3CCCC(O)C3)=O)C2)cn1 c1(CC(=O)NCC(C)NC(CSCC=C)=O)cc(F)cc2c1OCOC2 Cn1cc(Br)c(CC(=O)NC2CC2NC(=O)CCCn2cnc(C#N)n2)n1 N1(C(C2C(C)C2C)=O)CCC(CCNC(=O)C(C)Oc2cccnc2)CC1 C1(C(=O)NCCCN(C(c2ccc(C(F)F)s2)=O)CC)CCCN1C1CCCC1 N1(C(c2c(C)nc(O)[nH]2)=O)CCCC2(NC(C3CCSC3)=O)CC2C1 c1(CC(=O)N(C(CNC(c2n(CC#C)ccc2)=O)C)CC)ccc(OC)c(F)c1 C1(C(N2C(C)COCC2)=O)CC2CCC(C1)N2C(=O)C(C)(C)CN1CCCC1 N1(C(CN(C2CCC2)C(c2c(CC)nns2)=O)=O)CCOC(C(C)C)C1 CCCCC(O)CC(=O)NCC1CCC1C(N1CC(C(N)=O)C1)=O N1(C(=O)CN2CCN(CC)CC2=O)CCC2(CCN(C(c3cscc3I)=O)C2)C1 N1(CC)CCC(NC(C23CC(CNC(=O)C=C(C)C(F)F)(OC2)C3)=O)C(C)C1 N1(C(=O)NC(C)(C)C)CCCC(CSCC(=O)N(CC)CC)C1.C(=O)(C(C)SC)NC c1(CC)cc(C(N2CCCCCC2CNC(c2nc(C)n(C)n2)=O)=O)ccc1F N1(C(C(C(C)C)N(C)C)=O)CCC(C2CC2NC(=O)CC2CCOCC2)CC1 N1(C(=O)CCN2CCCC2)CC2(CCC(NCc3ccc(O)c(O)c3O)C2)C1 C=CCC(C)(O)C(=O)NC(C)CC1CN(C(=O)Cc2cc(Cl)cnc2C)C1 N1(C(C2C(CNC(C(N3CC(C)C3)C)=O)C2)=O)CCn2ccnc2C1C O=C(C1OCCc2c(Br)cccc21)NC(Cc1ccccn1)CO C1(C(N(CCOC2CC(SC)C2)C)=O)C2CCC(C2)C1NC(=O)C(C)(C)C C(C(=O)N=c1ccn(C2CCC2)[nH]1)=CC1N(C(C2(C)CCCN2)=O)CCC1 c1(C(=O)NCCC2CCN(C(CCCCC=C)=O)C(C)C2)ccsc1S(C)(=O)=O N1(C(C(C)n2ccnc2)=O)CC(N(C)C(c2cnn(CCF)c2)=O)C2(CC2)C1 c1(C(N2CCC(N(C(C(F)OC)=O)CCO)C2)=O)ccc(C(F)(F)F)c(C)c1 N1(C(CN(C)CC)=O)CC2CC1C2CNC(=O)C(C)(C)c1ccccn1 c1(C(=O)NCCC(=C)CNC(C2CN(C)CCO2)=O)cc(F)cc(C)c1N C#Cc1cccc(C(N2CCCCC2C(C)(C)CNC(=O)C2=C(Cl)CCC2)=O)c1 N1(C(C(CCC)CCC)=O)CC2CCC1C1CN(C(=O)CCP(C)(C)=O)CC21 c1(CCNC(N)=O)nc(C(c2ccccc2)OCC(C)(C)O)nn1-c1ccccc1 c1(CC(=O)NC23CCCN(C(C)=O)CC2C3)ccc2c(c1)ncn2C n1(CC)ncc(C(=O)NCC(C)(C2CC2)NC(c2cnc(Cl)[nH]2)=O)c1Cl C1(CC)CCCN(C(c2ccc(C(C)=O)o2)=O)C1C(=O)N(CCCC(C)C)C Cc1ccc(C(C2CC2)NCC2NCCC2c2ccccc2)c(C)n1 CCC(C(=O)NCC1COCCN1C(=O)CCc1ccc(Cl)cc1)C(C)(F)F C(=O)(C1=CCCCC1C)N(CC(=O)NCC(COC)(C)C)C(C)C c1(C(CC(=O)N(CC(C)NC(C2CC(C)(CC)C2)=O)C)C)ccc(F)cc1 c1(C(CN(CCCOCC(=O)NC2CC2)C)(C)C)cccc(F)c1Br C1(C(=O)NCC2CCCN(CC)C2)N(C(=O)Cn2ncnn2)CC12CCCC2 N1(C(c2ncn(C(C)C)c2)C(=O)NCC(F)F)CCCC1C1CCCCO1 C1(N(C(CC=CCC)=O)C)CCCC(NC(c2cc(CNC(C)=O)oc2C)=O)C1 C(=O)(C1=C(Cl)CC1)N1CC(N(C)C(c2coc(Br)n2)=O)C1 C#Cc1ccc(C(=O)NCCC2(NC(=O)CCNC(=O)NC)CCCC2)c(F)c1 N1(C(CN2C(C)CCC2)=O)CC(=O)NC2CN(C(=O)CN(C)CCO)CCC12 C(=O)(C(CN=[N+]=[N-])NC(=O)C(CCC)N(C)C)NC(C#C)CCC N(S(=O)(=O)N1CCCC1)c1nn(C)cc1Br.Cn1cnnc1S N1(C(C=C(C)C(F)F)=O)CCCC2(CCC(NC(c3cc(Cl)n[nH]3)=O)C2)C1 CCCCCC(CC)C(=O)N(C(C)CCNC(=O)CC1CC(C)(C)C1)C N1(C(=O)NCc2cc(C(F)(F)F)on2)C2CCC1CC1(C2)N=N1 N1(C(C2NC(=O)OCC2)=O)CCN(C(C2CC2c2ccccn2)=O)CC2(CC2)C1 C(C(CC(=O)NC(C)C(C)(C)OC)C1CCC1)NC(CC)=O.C1C(=O)N1 c1(C(=O)NCC2CN(C(c3c(C)[nH]cc3)=O)CC23CC3)cc2c(F)cccc2s1 c1(NCC2(C=C)CCC2)cc(NCC(c2ccccc2F)OC)ncn1 C(CC(=O)N(CC(C)C)C)N(C(C1C(C(=O)OCC)C1)=O)C(C)C C1(CNC(CC(C)c2ccco2)=O)CCCCC1N=c1[nH]nco1 N1CCCC(C)C1.c1(CC)noc(CCCOC)n1.c12noc(n1)C2 CCC(C)CCC(O)CC(=O)NC(C)(C)CNC(=O)C(F)C(C)C C(C(Cc1cnc[nH]1)C(=O)NCC1COCCOC1)NC(CSCCC#N)=O Cn1cnnc1CCNC(C1(CNC(=O)C(O)c2ccco2)CC1)=O N1(C(C2(SC)CC2)=O)CC2CN(C(c3ccc(N)cn3)=O)CC(F)(F)C2C1 N1(C(C2C(C)=C2)=O)CCC(C)(C)C(CNC(=O)Cn2nc(C)c(Cl)c2C)C1 C(CCS(N)(=O)=O)c1cn(CC(C)OC2CCOC2)nn1.C(=O)(C(F)OC(F)(F)F)N C(=O)(C1=NOC2(CCOC2)C1)NC1CCN(CCNC(CC(C)(C)C#N)=O)CC1 C1(C(=O)NCCn2cnc(C(=O)NCc3nnc(C)s3)c2)(CC)CCOC1 C1(C(=O)NCCCCO)CC2(CCN1C(=O)C1=CCOCC1)CC2 CCC(C(=O)NC(C)C(C)(C)NC(C1CCCN1C)=O)OC N1(C(COC)=O)CCOCC(CNC(c2ccc(-c3nnc(O)n3C)cc2)=O)C1 C1(CC(=O)NC23CC(CNC(=O)CCn4cncn4)(OC2)C3)CC(O)C12CCC2 C1(C=O)CC(F)(F)CN1C(=O)COC(C)(C)C.N12CC(C(C#N)C1)N2C c1(OC)c(C(=O)NCC(CNC(=O)CCC2CC2)OC)sc(C)c1Br C1(C(N2C(CN(C(c3c(SC)cccc3)=O)C)COCC2)=O)CC2CCC(C1)C2 C(CC(=O)N1CC(CC(C)C)C1)(C(C)OC)NC(c1ccn(COC)n1)=O c1(C(N2CCCCC2C(C)C)C(=O)Nc2c(CC)cccc2)ccc(Cl)c(Cl)c1 c1(OCC)c(C(=O)NC2CCC(NC(c3ccnc(C)c3N)=O)C2)cccc1F C(=O)(N=c1ccn(C)[nH]1)c1c(CNC(CSC)=O)nnn1C C(CS(=O)(=O)CC1CC(F)(F)C1)OCCC N1(C(=O)CCc2cccnc2F)CCC2(CCN(C(c3ccncc3)=O)C2)C1 Cc1cc2nc(C(=O)NCC3CCN3C(C3CC(C)(C)CO3)=O)cn2cc1C C1(NC(C2C(C)OC(C)C2)=O)CC2CCC1N(C(C1(OC(C)C)CCC1)=O)C2 C1(C(C(C)NC(=O)NCC2(N3CCOCC3=O)CC2)C)Cc2ccccc2C1.OCO C#CCCC(O)C(=O)NCCC1CSCCN1C(=O)COc1cccc(C#N)c1 C1(CNC(C(CC)CC2CCCCC2)=O)CCN(C(=O)C=CC(C)C)C12CCC2 C=CC(C)(CC)C(=O)N(C)CCN(C(c1nccc(OCC)c1F)=O)C(C)C c12ccc(c(F)c1)OCCOCC(=O)NC1CN(C1)CC(=O)N2.C1COC1.CCOC c1(OC)cccc(OC)c1C(=O)Nc1ccccc1-n1cc(C(C)OC)nn1 Nc1ccc(Cl)cc1C(N1CCCCC(NC(=O)Cc2cn(C3CC3)cn2)C1)=O c1(C(=O)NCCC2CCC(NC(C3(CCOC)CC3)=O)C2)cc(F)c(N)c(F)c1 c1(OC)cc(CN2CCCC(C(N3C4CCC3CC(O)C4)=O)C2)cc(OC)c1C C(=O)(CCCNC(c1c[nH]nc1C(F)F)=O)N(C)CC1CCCO1 CC(CC#N)C(=O)NCC1(CC(=O)NCc2cc(SC3CC3)no2)CC1 C1(NC(Cc2c(C)cco2)=O)CC(NC(C2(C)CCCS2)=O)C(O)C1 C(c1cccc(Cl)c1)=CC(=O)NC(CC(C)C)CNC(C1(F)CCOCC1)=O C1(C(N2CC(O)(C(C)NC(=O)C=CCF)C2)=O)CCC(C)(O)CC1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCC(NC(C(C)Cn2cccn2)=O)CC1 c1(C(=O)OC)ccc(C)nc1N(C1CCN(C(C2CCC(C)O2)=O)CC1)C C1(CC(=O)NCC(F)Cl)CC2CN(C(c3n[nH]cc3Cl)=O)CC2C1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CC(NC(C(CCCC)C)=O)C1 N1(C(CC2N(C(C3C(C)C3)=O)CCC2)=O)CCOC(C)(C2CC2)C1 C1(NC(Cn2cc(CNC(C3CCN(CCF)C3)=O)nn2)=O)CCCCC1CO N1(C(COC)=O)CCOC(C)(CNC(C2CCN(C(C)=O)CC2)=O)C1 C=CC1(C(N2CC(CCO)C2)=O)CCN(C(=O)CCCCCF)C1 C=C(C)C(C)(O)C(=O)N1CCC1CNC(c1ccccc1NC(=O)NC)=O c1(C(N(CCNC(c2cn(CCC)nn2)=O)CC)=O)nccnc1C(N)=O CN1CCN(C(=O)CC2CC(NC(C3OCCCC3(C)C)=O)C2)CC1C1CC1 c1(SC)ccc(OC(C)C(=O)NC(C)CN(C(=O)Cc2c(C)cnn2C)C)cc1 c1(C(=O)OC)c[nH]c(C(=O)N(C2CCN(C(=O)COCC(=O)NC)C2)CCO)c1 CCCC(CCC)C(=O)NC(C)(CNC(c1cccc(COC)c1)=O)CC(C)C c1(C(=O)NC2CCCN(C(=O)C(Cl)=CCl)CC2)nnn2c1CCCC2 c1(C2N(CC)CCC2)cccc(Br)c1.c12ccc(s1)CC(=O)N(C1(C)CCCC1)C2 C#Cc1ccc(C(N2CCC(C(=O)NCC(O)C3CC3)C23CC3)=O)cc1 C(C(CC(=O)NCC1CN(C)CCN1C(C1CC2CCC1O2)=O)C(F)F)N(C)C C(=O)(C(F)CC1CCCCC1)NCC1(NC(=O)NC2(C(=O)OC)CC2)CC1 N#Cc1ccsc1C(N1CCOC(C(N2CC(N3CCC3)C2)=O)C1)=O c1(NC(C2CCCO2)=O)c(C(=O)NCCCCOCCS)nnn1C.C1(=O)CN1.CS C1(c2cn(C)nc2)C2CCC(C2)C1N=c1[nH]nc(C2CCOCC2)s1 C1(CNC(c2c(COC)ncs2)=O)CCCCN(C(C2(C)CCCCC2C)=O)C1 C1(NC(C2(CC)CCOC2)=O)CN(C(=O)OCc2ccccc2)CC1N=[N+]=[N-] C=CCCCC(C)(C)C(=O)NC(CNC(c1cc(O)ncn1)=O)CO C1(C(N2CC(CNC(=O)C(C)(C)CO)C(C(F)(F)F)C2)=O)(OC)CCC12CCC2 C(=O)(C1=CCC(C)CC1)NC1(C(=O)NC2C(COC)CC2)CC1(C)C C1(CNC(C2(C)CN(C)C(=O)C2)=O)CCN(C(c2sccc2F)=O)C12CCC2 c1(C(=O)NC2(CC(=O)OC)CC2(F)F)cc(C)ccc1Br C12(CNC(C3CCCN(C(=O)OC)C3)=O)CN(C(=O)CCCC3CC3)CC1CCO2 C1CN=C(NC(C)C(c2ccccc2)C)NCc2cnc1cn2.CO C1(NC(CSCCN(CC)CC)=O)CCC1NC(C1(C(=O)NC)CC1)=O CCC(CC)C(C)C(=O)NC1CC=C(C(=O)NCC(CC2CC2)CO)C1 CCC(C)CCCCC(=O)NCC1CN(C(c2cc(C#N)ccc2F)=O)C1 N1(C(C(c2ccccc2)OC(C)C)=O)CCCN(C(C2CCCOC2)=O)C(C)C1 CCCC(C(=O)NCCOCCC(=O)N1CC(N2CCCCC2)C1)OC C1(N(CC)CC)CCN(C(c2ccn(C(C)C)n2)C(=O)NCCSCC#N)C1 C(=O)(CC(C(F)F)NC(=O)CC1CCC(=O)C1)NC(c1nc(C)[nH]n1)(C)C CC1(C)CC(=O)N(CC(N2CC3(NC(=O)C=Cc4ccc(CO)o4)CC2C3)=O)O1 CCC(C(=O)NCC(C)N(C(=O)C=CC(=O)OC(C)(C)C)C)C(C)(F)F CCCCCCCCC(=O)Nc1cccc(F)c1F CC(C)C(O)(C(=O)N1CCN(C(=O)CCc2nc(O)n[nH]2)CC(O)C1)C(F)(F)F C1(NC(CCC)=O)CCC(C)N(C(=O)C=CCN2CCCC2)C1 C(C(C)(C)C(=C)C)N(C(=O)Cc1ccsc1)CC#C.C(C(=O)N)=C c1(C(=O)NC2CN(C(c3c(C)onc3O)=O)C2)cc(Cl)c(Cl)cc1N N1(C(CNS(CCCC)(=O)=O)=O)CCC(NC(=O)CCC2CCOC2)CC1C c1(OCC(=O)NCCn2nnc(C)n2)cnc(C)c(C(=O)O)c1 c1(C(CNC(c2ccc(C(C)=O)[nH]2)=O)NC(C2(C)CCCC2)=O)ccc(F)cc1 C(CC(C(=O)NC1(C(=O)NCc2onnc2C2CC2)CC1C)OC)OC N1(C(COc2ccc(C)cc2)=O)CCC(NC(c2cscc2Cl)=O)CC1C Cn1c(C(N2CC(NC(=O)CC3CCC(C)(C)O3)C(C)(C)C2)=O)cnc1[N+](=O)[O-] C=CCC(CC(C)C)C(=O)NC1(C)CN(C(=O)CCc2cc(C)n(C)n2)C1 C1(NC(N2CCN(C(=O)C(F)F)CC2)=O)CC2(CCCC(CO)O2)C1 C(C(CNC(=O)CCSc1nnnn1C)C(F)(F)F)NC(CC(=C=C)C)=O C=C1CCN(C(C2CCC(=O)C2)=O)C(C(=O)NCC2(CN(C)C)CC2)C1 C1(CNC(C)=O)CCCN(C(=O)NCc2cccc(Br)n2)C1 C1(NC(c2c(C)nc(CC)s2)=O)CC2(NC(C3CCN(C)C3=O)=O)COC1C2 N1(C(C2C(C)(C)CO2)=O)CC(CNC(=O)C(F)n2ccnc2)CC(C)(C)C1 C1(C(C)C)C(NC(=O)CCCc2cccs2)CCN1C(c1cnc(C2CC2)s1)=O N(C(=NCCCCl)NCc1c(C)cccc1Br)C1CC(OC)C12CCC2 N=c1[nH]nc(C(N2CC(CC(F)C(=O)NCC3CSC3)C2)=O)[nH]1 S(=O)(=O)(c1ccccc1)NC(CC(=O)NC(c1ccc(O)cc1)C(F)(F)F)=O c1(C(=O)NC23CC(NC(c4cnco4)=O)C(OC2)C3)n[nH]c2c1CCCC2 Cn1cc(C(=O)NC(C2CCCC2)CNC(=O)COC2CCOCC2)nn1 Cn1nnc(C(=O)NC2CC2NC(=O)CCc2cc[nH]n2)n1 Cc1ccc(C2CC2)cc1C.C1(=O)C(C)(c2ccccc2)CSCCC(=O)O1 Cc1ccc(OCCC(=O)NC2CN(C(c3cccnc3)=O)CC2C)c(C)c1 c1(C(CNC(C2CC2(Cl)Cl)=O)NC(COC)=O)ccc(C)cc1.C12CC(C1)N2 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(=O)COc2cccc(F)c2)CCC1F n1(-c2cccc(C(=O)OCC)c2)cc(C#CCN(C(c2cn[nH]c2)=O)CC)nn1 CC1=C(CNC(=O)CCC2CCCN(C(c3cc(C)c(C)s3)=O)C2)COCC1 c1(OC)ccc2nc(CNC3(N)CC4CCC(C4)C3)[nH]c2c1 N1(C(C2CCC2)=O)CC2CCC(C1)N2S(=O)(=O)CCC(F)(F)F.C1CCC1 c1(NC(c2ccc(-c3n(C)ccc3)c(F)c2)=O)cc(F)c(F)c(F)c1F N1(Cc2cn(C)nc2Br)CC2CCCCCC2C1 C(=O)(CC1=CCN(C(=O)C2CC2)CC1)NCC(N1CCCC1)C C(N=c1[nH]cnc2ccc(O)cc12)C1CCC(NC(c2n[nH]c(C)c2O)=O)C1 N1(C(C(C(=C)Cl)(C)C)=O)CCC(F)(F)C(CNC(=O)CC2CC2CC)C1 N1(C(c2nsc(NC(C3C(C(=O)OC)C3)=O)c2Br)=O)CCC2(CCCO2)C1 CCCCCC(C)CC(=O)N1CCC(CCC(N2CC3C(CO)C3C2)=O)CC1 C(=O)(C1CC(O)c2ccccc21)N1CC(C)(NC(=O)Cc2ncc(Br)s2)C1 CC1=C(C(=O)NC2CCC(C)(C)CC2CNC(C2(C3(C)CC3)CC2)=O)COCC1 C1(CNC(c2nc(C)sc2)=O)CC2(CCC2)CN1C(=O)C(C)Oc1ccccc1 c1(NC(=O)COC(=O)CCCc2ccccn2)ccccn1 C1(NC(c2c(Cl)cc(C)s2)=O)CC2CC(C1)N(C(c1nccn1C)=O)C2 C1(n2cc(CCNC(N(C)C)=O)nn2)CON(C(=O)c2csc(O)n2)C1 c1(C(=O)NCC2C(CNC(CC3(CS(C)(=O)=O)CC3)=O)C2)c(N)sc2c1CCC2 N1(C(C(COC)(C)C)=O)CCC2(COC(CNC(c3conc3C(C)C)=O)C2)C1 N1(C(C2C(CCC)CCC2)=O)CCC(F)(F)C(CNC(c2nc(O)sc2C)=O)C1 C=CCC(C)(C)C(=O)NCC(CC(F)(F)F)n1cc(C(C2CCOCC2)C)nn1 C1(NC(C(C)Sc2nncn2C)=O)CCN(C(c2ncn(C)n2)=O)C12CCC2 CN1CC2(CN(C(=O)C(c3ccoc3)NC(=O)CNc3ccccn3)C2)C1 c1(NC(CNC(c2n(CCC)ncc2)=O)(C)C)nc(C(=O)OC)c(C)c(C)n1 c1(C(=O)NC(CCOC)CNC(c2cccc(OC)n2)=O)ccc2n[nH]cc2c1C O(N1C(=O)c2ccccc2C1=O)CC(=O)NC(C(C)NC(=O)C(=O)NC1CC1)C c1(C(=O)NC2CC(C)N(C(=O)CCc3nc(O)n[nH]3)C2)cnc(Br)c(N)c1 c1(OC)ccc2c(c1)CN(C(C1CC1c1c(F)cccc1Br)=O)CC2=O N1(C(C2CC(OC)C2)=O)C(CC(=O)NC2CC23CCCC3)C2CCCC12 C1(CC)(CO)CCCN1C(=O)NCCN1CCC(OC(C)=O)CC1.C(C(F)(F)F)O C(=O)(C(CC(C)C)C(C)C)N1C(CNC(=O)C2=NOC(C)(C)C2)CC(OC)C1 C1(OC)CN(C(c2nccn2C)=O)C(C)(CNC(=O)CO)C1 c1(C(=O)NCCN(C(C2CCC(=O)NC2)=O)C2CC2)cc(F)ccc1F c1(OC)cccc(CC(O)C(=O)NC2CC2NC(c2ncccc2C(F)F)=O)c1 Cc1ccc2[nH]c(C(=O)NCC(C)CNC(=O)C(c3ccncc3)C)c(C)c2c1 C1(CC(=O)NC(COC)C(=O)OC)CN(C(=O)Cc2ccsc2C)CCC1C c1(C(=O)NC2CCN(C(C(CCCC)C)=O)C2(C)C)cc(C)nc2ncnn12 c1(C2N(C(C3CC(NC(C(C)SCCCC)=O)C3)=O)CC2)cccnc1 C1(CNC(CCC(C)(C)OC)=O)CCC2(CCC2)C1NC(c1nnccc1C)=O Cc1cc(C(=O)NC2CC(CNC(C3CC=CCO3)=O)C2)ncc1S(N)(=O)=O C1(NC(C2(C(C)C)CCC2)=O)CCCC(NC(c2cn(C)ccc2=O)=O)CC1 N1(C(c2ccncc2Cl)=O)CC2CCN(Cc3c[nH]c(Br)c3)C2C1 c1(C(N(C2CCN(C(=O)C(F)C3CCC3)CC2)CC)=O)c(Cl)nc2ccccn12 C(=O)(CC(O)CCNC(=O)C(F)(F)C(C)O)N(CCCN(CC)CC)C C(=O)(CC(C)(C)C(=O)N1CC2C(C(=O)NCC(F)CO)C2C1)OC O=C(C1=CC2(CCOCC2)C1)NCC1CN(C(=O)C2=CCCS2)CCC12CCC2 C1(C(N2CCC(O)C2)=O)(CC)CCN(C(=O)C(SC)SC)C1 c1(CC(=O)N(C2CCCN(C(c3cnnn3CC)=O)C2)CC)cccc(Cl)c1 C(=O)(CCCCCCNC(=O)C(c1cnn(C)c1)=O)NCC(C)CN(C)C Cc1ccc(C(=O)NC(C)CC(C)NC(c2ncc(-c3ccccc3)o2)=O)s1 N1(C(c2ccc(CCC)cc2)=O)CCN(C(=O)C(O)CF)CC(O)C1 N1(C(CNC(N)=O)=O)CCC(O)(Cc2cn(CC3CC4C=CC3C4)nn2)CC1 c1(C(N2C(CN(C(CC=CC=C)=O)C)CCCC2)=O)ccc(C)cc1NCC C1(CNC(CNS(CC)(=O)=O)=O)CC(C)N(C(C2CCCO2)=O)C1 N(C1CCCc2ccc(Cl)cc21)C(c1cc(C)c(C)s1)c1nnnn1C1CCC1 Cc1ccc(-n2cc(NCC(CO)NC(=O)Cc3nnc(C)n3C)nn2)cc1 CCC(CC(=O)N1CCOCC1CN(C)C(C1CN(C)C1)=O)C(C)(C)C CCC(C)CCC(=O)NCC1CC(C)N(C(=O)Cc2ccc(F)nc2)C1 c1(C(=O)NCc2oc(C)c(C(=O)NC3CC4CCCC4C3)n2)cccc2cc[nH]c12 C1(NC(c2c[nH]ccc2=O)=O)CCCCC1C(=O)NCC1CCCOCC1 C1(C(=O)NC2C(CNC(c3c(CC)c[nH]c3)=O)CCC2)CCCCC12CCC2 c1(NC(C2CCCN(C(c3ccc(S(C)=O)cc3)=O)C2)C)ccnc2ncnn12 c1(OC)ccnc(C(=O)NCC2CN(C(=O)C(C)(C)c3ccsc3)CC2C)c1O C1(CNS(c2cc(OC)ncc2)(=O)=O)CCc2c(ncn2C)C1 C=CCC(C)C(=O)NC1CN(C(C2CC2NC(=O)OC(C)(C)C)=O)CC1F C1(C(N)=O)CCCCC1C(=O)NC1CC(CCNC(c2n[nH]cc2Cl)=O)C1 c1(C(N(CC(CC)NC(c2ccn(C3CC3)n2)=O)C)=O)ccc2snnc2c1 C1(CNC(c2ccc(CNC(C3(CCCC)CC3)=O)o2)=O)COCC(C)O1 CC1=CCCN(C(=O)CCC2CCCN2C(c2cccc(CN(C)C)c2)=O)C1 Cn1nc(C(=O)NC2(CNC(=O)CN3CCCNS3(=O)=O)CCC2)c2c1CCC2 c1(C(C(=O)OC)=O)ccnc(NNC(=O)C2Cc3ccccc3C2)c1 c1(CC)ccccc1-c1cn(C2CCC(C(=O)N(C)Cc3cccnc3)C2)nn1 c1(OCC(N)=O)ccccc1C(N1CC2CC2(NC(=O)C2=CCC2)C1)=O CC(C)(C(F)C(=O)N1CCCC(CO)(NC(=O)COC2CC2(F)F)C1)C(F)(F)F C1(N(C(c2c(C)nc(O)[nH]2)=O)C)CCCCN(C(C2CC(C)CC(=O)N2)=O)C1 C1(NC(C2CC(CC)(CC)C2)=O)CCCCC1NC(c1ccnn1C1CCC1)=O C(CC(CNC(C1COCCO1)=O)NC(=O)COCc1ncnn1C)OC N1(CC)CCCC1C1CCCN1C(=O)C(=O)Nc1ncccc1Br N1(C(CN2C(=O)CCC2)=O)CCC(CNC(=O)Cc2ccccc2)C(O)C1 C1(CNC(c2c(CC)ccs2)=O)CN(C(c2cc(COC)no2)=O)CC(C)(C)O1 C1(CNC(c2nnn(C)n2)=O)C2CN(C(c3cc(O)ncn3)=O)CC12 C1(C(C)(C)NC(C(C)(F)F)=O)CCN(C(c2ocnc2C2CC2)=O)CC1 N1(C(C)C)N=C(C(=O)NC2CC23CCN(C(C2CC2C#N)=O)CC3)CCC1=O CCC(CC)C(C)C(=O)N1CCN(C(c2cccc3nncn23)=O)CC1C C1(CNC(C=CC2N(C(CCOCC(C)C)=O)CCC2)=O)CN2CCC1CC2 C1(c2n(C)ccn2)CN(C(C2(SC3CC3)CCC2)=O)CC1NC(=O)C(O)C1CC1 C(N=C(NCC(F)F)NC1CC2(CCC2)OCCO1)C1C(C)(CC)C1 c1(C(=O)OC)cc(Br)c2nc(N)sc2c1.C(CCO)NC(=O)N(C)CCO c1(C(N2CC(CNC(c3cc[nH]c3)=O)OCC2)=O)ccc2c(c1F)CCC2 Cc1cc(C(N2CCC(C(C)(C)C)(CNC(C3CCCN3C)=O)C2)=O)nc(O)n1 CCC(CC(=O)N1CC(C(C)NC(=O)C(C(C)C)SC)(COC)C1)C1CC1 N1(C(c2nn(C)c(=O)cc2)=O)CC2CN(C(C34CCCCN3CCC4)=O)CC2C1 c1(C(N2C(C(N(C3CCC3)C)=O)C=CCC2)=O)c[nH]c2cnccc12 c1(OC)cccc(C(=O)N(CCN(C(=O)C(c2ccccc2)F)C)C(C)C)c1C c1(CC(=O)NCCC2CN(C(C3CCC(C#N)C3)=O)C2)ccc(O)c(F)c1 C(c1cccnc1C)=CC(=O)NCCNC(c1n(CC)ccn1)=O Cn1ncc2c(NCc3cc(C4CC4)no3)nc(N3CCC(CO)CC3)nc12 C1(CNC(C(C)NC(=O)C(N2CCSCC2)C)=O)CCCCN1C N1(C(=O)C2CC2)CC(NC(C2CC(F)C(=O)N2Cc2ccccc2)=O)CC(O)C1 C12(C)CCN(C1)C(=O)OC2.C(CC(=O)O)NC(C)C.C#CCCC=O c1(C(N2C(C)CC(NC(=O)C=CC(=O)N(C)C)CC2)=O)cc2cc(C#N)ncc2[nH]1 C(=O)(C(C(C)(C)C)C1CCCC1)N(CCCNc1cc(C)c(C)o1)C C1(C(=O)NC2(CSC)CCC2)CN(C(=O)C2=NOC(C)C2)CCN1C c1(NC(=O)NC(c2ccc(C)cc2)C=C)ccc(OC2CCC2)cc1 N(C(=NCC1CCOC(C)C1)N(C)Cc1cnn(C)c1)Cc1c(C)ccs1 C1(NC(Cc2cccc(COC)n2)=O)CN(C(=O)CC2(C)CC2)CC(C)(C)C1 C1(C(=O)NC2(C3N(C(C(C4CCS4(=O)=O)=O)=O)CCC3)CC2)C2CC3C(C2)C13 c1(C(=O)NCC(CCOC)NC(=O)C(C#N)C2CC2)ccc(OCC(N)=O)cc1 C(N=c1[nH]ncs1)C1C(C)C1.N12CCC(C1)C2C(=O)NC1CC(F)(F)C1 CCCCC(F)(F)C(=O)NC1COCCN(C(=O)CCc2nnc(C)n2C)C1 C(Cc1ccccc1)(C(=O)NC1CCCC1OC(C)(C)C)OCC Nc1cccc(C(=O)NC2CC2NC(c2cncc(OC3CC3)c2)=O)c1 C(CNC(=O)C(O)C1(N(C)C)CC1)(CCNC(=O)CCOCCF)OC C1(C(=O)NC2CN(C(c3cc(O)ncn3)=O)CC2CO)CC12CCCCC2 NC(=O)CCCCC(=O)NC1CCCN(C(c2c(O)ncc(Br)c2C)=O)C1 c1(C(=O)NCC(C)(C)NC(=O)CC(O)c2ccccc2)ccc(P(C)(C)=O)o1 CCCC(O)C(=O)NC(C)CCNC(=O)Cc1csc(Br)c1 Cc1cc(N)c(C(=O)NC2CC2CNC(=O)CCCCCNC(N)=O)cc1C C12(NC(=O)CC3CCC3)COC(C1)C(NC(c1cnn(-c3ccccn3)c1)=O)C2 c1(OC)cncc(C=CC(=O)NCC(C2CC2)NC(=O)Cc2ccccc2C)c1 c1(COC)nn(C)c(Cl)c1C(=O)NCC(CO)NC(=O)C=CCO C1(C)(NC(C(C2CCOCC2)OC)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1 C(CCNC(C1(NC(=O)Cn2cncn2)CC1)=O)(C(C)C)OC N1(C(Cc2n(C)ccn2)=O)CC2C(CNC(C3(c4ccc(F)cc4)CC3)=O)C2C1 CCC(C)CC(C)NC(=O)CN(C1CC(C#N)C1)C(c1cc[nH]c1)=O CC(C)CCC(=O)C(=O)N1CC(C(N)=O)(CNC(=O)CCc2ccsc2Cl)C1 C1(C(C)C)CN(C(c2cc(Br)ccc2Cl)=O)CCN1C(=O)C(C)CF N1(C(C2N(C(c3nc(CC)oc3)=O)C(C(C)C)CC2)=O)CCN(C2CC2)C(=O)C1 N1(C(CNC(C(C)C)=O)=O)CC2C(CNC(=O)CN3CCCCC3)C2C1 C#Cc1ccc(C(=O)NCCN(CC(C)O)C(C2CC(C3CCC3)C2)=O)cn1 N1(C(C2C(C)C2)=O)CC23CCCCC2(C1)CN(C(C1CCCCC12CCC2)=O)C3 N1(C(CN(CC(C)C)C(=O)CC2CCCOCC2)=O)CCN(C)CC1CCO N1(C(c2ccn(C(C)C)n2)=O)CCCC(C)C1CNC(=O)CCc1cccn1C c1(CN(C2CN(C(=O)C(F)C3CCC3)C2)C(=O)C=CC2CCC2)ccccc1 C1(CC(=O)NCCOCCCNC(c2c(OC)csc2)=O)CC2C=CC1C2.C(=O)N c1(C(N(C2CCN(C(=O)CCSCC)CC2)CCC)=O)cc(F)cnc1O C1(CNC(c2ccc(C)nc2)=O)CCN(C(=O)CCc2cccc(Cl)c2)C(C)C1 c1(CCC)c(C(=O)NCC(C)(C)CCNC(=O)CC2CC3C=CC2C3)nnn1C N1(C(CC(CC)O)=O)CCC(C(=O)NCCOC(C)C)(OC)CC1 c1(C(N2C3CC(NC(=O)Cn4cnnc4O)C(C3)C2)=O)n[nH]c2c1C(=O)CCC2 c1(NC)ccc(C(=O)NCC=CC(=O)Nc2ccnc(C3CCC3)c2)cc1 CC(C)CC(C)(O)C(=O)N1CC(C(=O)NC(c2cscn2)CO)C(F)(F)C1 c1(C(=O)NC2C(C=C)CN(C(=O)C(C)C(C)C)C2)cc2c(nc1O)CCC2 C1(CCNC(C2CCOC2)C)COC(C)(C)OC1 C(=O)(C(F)CC(C)(C)C)N1CCC(NC(c2c(C(C)=O)cccc2)=O)C(O)C1 Cc1cnn2cc(C(=O)NC(C)(CNC(c3ncncc3Cl)=O)C3CC3)cnc12 N1(C(C(CC(C)C)C)=O)CCN(C(c2cn(CC(F)F)cn2)=O)CC(CO)C1 C1(C(=O)NCCCN(CC(C)C)C)CCN(C(=O)Cn2cncn2)CC1(C)C C(=O)(CC(C(=O)NCC1CCCC(NC(c2cnc(C)[nH]2)=O)C1)N(C)C)OC CC1(C)CCCCC1C(=O)NCC1C(CNC(C2CC(F)(CF)C2)=O)C1(F)F Cc1cc(NC(C2CCC3(CC3)N2C(=O)CSC(F)F)=O)c(C)c(C)c1 C1(C)(C(=O)NCC(CC)NC(=O)C(c2nncn2C)c2cccs2)CCCCO1 c1(-n2ncc(C(=O)NC(C)CCNC(=O)C=CBr)n2)ccc(Br)cc1 C1(CC)CCC(N(C(=O)CCC(C)NC(c2cccc(O)c2)=O)C)CC1 c1(C(=O)OC)cncc(C(=O)OCC(C)(C(F)(F)F)c2ccccc2)c1 Cc1cccc(F)c1C(=O)N(CC(C)C(N1CCCC(N(C)C)C1)=O)C1CC1 c1(OC)cc2ccc(CNCC3CCCN(CCC#N)C3)nc2cc1F CN1CC2(CCN(C(C34CC(C(=O)O)(C3)C4F)=O)C2)OCC1=O Cc1cccc(C)c1NC(=O)C(c1cc(Br)no1)N(C)Cc1nccs1 Cc1cc(NC(CN(C)CCOC(C)(C)C)=O)c(C)n1-c1ccccc1 C1(C(C2CC2)NC(C2CCCO2)=O)CCN(C(=O)CC2CSC2)C1 Cc1c(C(N2CC(C(N)=O)(CNC(=O)CCC3CCCO3)C2)=O)ccn1CCO C12(C(=O)NCC3COCCN(C(CCC(=C)C)=O)C3)CCCCCC1OCC2 C1(NC(C2CCC(CNC(Cc3c(C)nn(C)c3)=O)O2)=O)CCC(=O)NC1C c1(C(=O)NCCN(CC(C)O)C(c2ccccc2)=O)c[nH]nc1C1CCOC1 CC1CN(C(c2ccncc2O)=O)CCCN1C(=O)CC12CC(C1)C2 n1(CCC(N2C(CCNC(C(C)SC)=O)CSCC2)=O)ccc2cc(Cl)ccc12 Cc1cccc(OCCCC(=O)N2CCCC2C2CC2)c1.C(=O)(CCCN(C)C)NC N1(C(C(Cc2ccccc2)OC)=O)CCC(NC(=O)CC2CC2C)C(C)(C)C1 c1(C(=O)NC2C(CNC(CCC(=O)NC)=O)CCCC2)n[nH]c2c1CC(C)CC2 N1(C(COC(C)(C)CN(C(=O)Cc2ccco2)C2CC2)=O)Cc2ccccc2C1 C12(C(=O)NCO)OC(C(F)(F)F)(C1)C2.C12(C#N)CC1N(C)CCOCCNC(=O)C2 C(=O)(CS(=O)(=O)NCC1CCCCO1)NCC1N(C(C2CCCC2)=O)C2C(C1)C2 CCC(CN(C)C)CC(=O)N1CCC(CCNC(c2cnsn2)=O)C1 C1(C2N(C(CCc3c(C)ncs3)=O)CCC2)CCN(C(C2CC23CCC3)=O)CC1 Nc1ccc(CCNC(N2CCCCC2CSc2ccc(F)cc2)=O)cc1 c1(CC(N2CC3C(NC(c4c(CC)scc4)=O)C3C2)=O)ccc2c(c1)CCOC2 C1(C(=O)NCCc2cncc(C)n2)(CC)CCCN1C(C1CC=C(C)CC1)=O C(=O)(CC(CN(C)C)C(F)(F)F)N1C2C(NC(c3ccc(OC)o3)=O)C(C2)C1 C1(c2cccnc2)(C(N2CC(NC(C3(CCO)CC3)=O)C2)=O)CCCCC1 C#Cc1ccc(C(N2CCC2CC(=O)NCCn2cccn2)=O)cc1 N1(C(CC=C=C)=O)CCCC1(C)CNC(=O)C(C)Cc1ccccn1 C=CCCCCC(=O)N1CC(NC(c2ccc(NS(C)(=O)=O)nc2)=O)CC1CO Cc1cc(Cl)ncc1CC(=O)NCCCCNC(c1ccc(F)c(C)c1)=O CON1CCC(N(C)C(C2CCN(C(c3ccc(=N)[nH]c3)=O)CC2C)=O)CC1 N1(C(CCSC)=O)CCC2(NC(C34CC(C(C)(F)F)(C3)C4)=O)CC2C1 c1(NC(N2CCCC(C(=O)OCC)C2)=O)ccc(NC(c2ocnc2C)=O)cc1 C1(C)(C(N2CCC(C)(CSC)C2)=O)CCCN(C(=O)C(C)CCCOC)C1 C1(C(=O)OCC)CCOCCN1C(c1cc(-c2ccc(C)cn2)on1)=O Cc1nc(C(C)C)oc1C(=O)NCC1CCCCN1C(c1cc(Cl)ccn1)=O C1(C(N2CC(N(C(=O)C(C)CSC)C)C2)=O)(OC)CC1(F)F C(=O)(C1Cc2ccc(F)cc21)NCC1CN(c2nc(C)c([N+](=O)[O-])cn2)C(C)C1 C(=O)(C1=CC2(CCOCC2)C1)N1C2CCN(C(c3cc(CC)no3)=O)CC2C1 O=C(CCCCCC1CCc2ccccc21)NCCC1CCC2(CC1)OCCO2 c1(N)cc(F)c(F)cc1Cl.c12cc(ncn1)N(C1CCNCC1)C(=O)N2C(C)C C1(CCNC(=O)CSC2CCCCO2)CCCCN1C(C1CC2(CSC2)C1)=O C1(NC(C(C)NC(N)=O)=O)CCCN(C(=O)C=Cc2cncc(F)c2)CC1 N1(C(CC(C)F)=O)CC2(C1)CN(C(=O)C1=CC3CCC(C1)C3)CCO2 Cc1ccc(F)cc1C(=O)N(C(C)(C(=O)NC1CCCC(O)CC1)C1CC1)C C(CN=C(NCC(F)(F)Cl)NC1CCN(c2nc(C)cs2)CC1)SC C=CC1CCC1C(=O)NC12CC(CNC(=O)CCc3ccccc3)(C1)C2 Cc1cc(Cl)cc(C(=O)NC(C)CCNC(=O)Cc2n[nH]cc2Br)c1N C1(C(N2CCN(C(c3ccc(Br)cc3)=O)CC2)=O)CCn2c(Br)cnc2C1 c1(C(N(C(C)C)CCN(C(=O)CSC(F)(F)F)C)=O)ccccc1C1CCC1 CCCCCCC(=O)N1CC(NC(C2CCCCC(=O)N2)=O)C2CC2C1 C1(CNC(c2ccc(Cl)cc2Cl)=O)CCCCN(C(=O)CSC2CC2)C1 C(C(C)(C)C#CC(=O)N(CC)CC1CCCO1)NC(C1CC(C)(CC)C1)=O C1(C(=O)NCCN(C(c2ccc(CSC)o2)=O)C2CC2)CNC(=O)CC1C CC(C)(CNC(C1CCC(=O)O1)=O)CC(=O)NCC1CC1c1ccco1 c1(C(=O)OC)cnc(N2CCN(C)CC2CNC(c2cocc2C)=O)cc1C Cc1nsc(C(N2C(CNC(=O)CN(C3CCSC3)C)CC3CC23)=O)c1N N1(C(=O)CCc2cccc(F)c2)CCC2(C1)CN(S(=O)(=O)c1ccc(Cl)s1)C2 c1(C(N(CC(C)NC(C=CCC)=O)C)=O)cccc(-c2ccccc2)n1 CC(CS(C)(=O)=O)C(=O)N(CC(=O)OC)Cc1cn(-c2ccc(Cl)cc2F)nn1 c1(C(c2nnnn2-c2ccccc2Cl)NCCOC)cnn(C(C)C)c1C c1(C(=O)NC2(C)CN(C(C3CC3c3ccco3)=O)C2)sc(Cl)cc1Cl C1(C)(C(N2C(COC)CC(O)C2)=O)CN(C(=O)CC2COC(=O)C2)CC1C N1(S(c2cc(C)sc2)(=O)=O)CC2CCN(C3CCCC3)CC2C1 N1(C(C(C)(C2CC2)OC)=O)CCN(C(C2(n3cncn3)CC2)=O)CC12CCC2 c1(C(N(CCCC(=O)NC(C2CCOC2)CC)C)=O)ccnc2cc[nH]c12 C(CC(=O)NC1CC1NC(=O)C(O)C1CCCC1)SC N1(C(C2CCC(C)C2)=O)CCOC2(CCC(NC(=O)C3=CCOCC3)CC2)C1 c1(N(CCCNC(=O)C(C)NC(N)=O)CC)cc(-c2cccs2)nc(Cl)n1 C1(OC(C)CNC(C)COc2ccc3c(c2)OCO3)CCCC(F)(F)CC1 Cc1cc(CNC(C2CCN(C(=O)C=Cc3ccoc3)C2)=O)n[nH]1 C1(C(N2CCC(CCNC(CC=C(C)C)=O)C2)=O)OC(C)(C)OC1(C)C c1(C(=O)NC2CN(C(c3n(CC)ncc3)=O)CC2C)c(F)cc(F)cc1Cl c1(C(=O)NCC(CC(C)C)NC(CCc2cc(C)no2)=O)c(Cl)nn(C)c1Cl C1(CNC(=O)CSCc2ccccn2)CCC(NC(C2(CCO)CC2)=O)CC1 N1(C(Cn2nnc(=N)[nH]2)=O)CC2(CCC(CNC(=O)Cc3ccco3)O2)C1 C1(C)(CNC(c2cn(CC=C)nc2)=O)CN(C(c2ccc(C#N)s2)=O)C(C)(C)C1 c1(OC)cccnc1NC(c1cc(C(F)(F)F)sc1C)=O c1(CNCCOC(C)(C)C)cc2ccnc(F)c2o1 C(=O)(C1CCCc2ccnn21)NC1CC2CN(C(CCC)=O)CC2C1 CC(=O)CC(C)(C)C(=O)NC(C)C=CC(=O)NCC1CC(O)C1(C)C C(=O)(C1=CC2CCCCCC12)N(CCN(C(c1c(CC)cco1)=O)C)C(C)C c1(C(N2CCC(NC(C(CC)OCC)=O)C2)=O)cnc2[nH]ccc2n1 c1(C(C(=O)OC)N(C(C2(CC)CC2)=O)CC2CCOC2)noc2c(Cl)cccc12 C1(CCNC(c2ccc(CCF)cc2)=O)CCCN(C(=O)C(O)C2CC2)C1 Cc1ccc(F)c(C(C)NC(N2CCCC23CNC3)=O)c1F Cc1cc(C(N2CCCC2c2csc(C)n2)C(=O)NCCCF)cc(F)c1 c1(C(N(CCC)CCNC(=O)CCN(CC)CC)=O)c2c(c[nH]c1=N)CCC2 C(=O)(C1=CCCCC1)NCCCC1CCCN(C(C2CCOC2C2CC2)=O)C1 N1(C(CCN(CC)CC)=O)CC(OC)C(NC(=O)CCC2CCCOC2)C1 C(=O)(C1=NOC2(CCOC2)C1)N(CCNC(c1c(C)cc[nH]1)=O)C(C)C N1(C(C2C=CCC2)=O)CCC2(CC1)CCN(C(C1CC(CC3CC3)C1)=O)C2 C1(C(=O)NCC2C(CNC(C(C)(Cl)Cl)=O)C2)CC12CCOc1ccccc12 c1(C(=O)NCc2cc(C(=O)N(C3CCOC3)C3CC3)on2)cnc(Cl)cn1 c1(NC(CC(C)NC(=O)C(C)(C)CO)C)ncc(C#N)cc1F C(=O)(CC1OCCc2ccsc21)NCCCC(c1ccccc1)NC(C=CC)=O CC(C)(O)C(F)C(=O)NCCN1CCN(C(C2(C)CC(C#N)C2)=O)CC1 N1(C(c2c(CC)ncnc2)=O)CC2CC(NC(=O)CCSc3ccccc3)C1C2 Cn1nnc(Br)c1C(=O)NCCC1CCCN(C(C2CS(=O)(=O)C2)=O)C1 c1(C(N2CCCC(NC(c3ccc(Cl)s3)=O)C2)=O)cnc2[nH]ncc2c1 C(C1c2ccccc2CCN1C(=O)CC(C)OC)NC(CC=C=C)=O C(C1CCCO1)=CC(N1C(CNC(C2CCCCS2)=O)CC1)=O C(=O)(C(C(C)C)c1ccnc(O)c1)NCC1(NC(C(C)SCC)=O)CCCC1 Cn1ncc(C(=O)NC2(C(=O)NCC(C)(O)C3CCC3)CC(O)C2)c1Cl CC(C)C(F)(CNC(=O)CSC(C)(C)C)C(=O)NCC1CN2CCC1CC2 c1(C(=O)NCC2CN(C(Cc3cc(C)ns3)=O)C(C)(C)C2)cn2cccnc2n1 c1(C(=O)NCC2(OC)CN(C(C3CC(C)CO3)=O)C2)cnc(NC(C)=O)cn1 c1(CC(=O)NCCN(C(c2cnc(-c3cnn(C)c3)s2)=O)CC)nc(C)c(C)o1 C(=O)(CCCCCOC)NC(CNC(C(c1cccc(C(=O)OC)c1)(F)F)=O)C C1(NC(=O)CC23CC(C2)C3)COCC1CNc1cn(Cc2cccnn2)nn1 N1(C(c2c(C)nc(C(C)C)s2)=O)CC(CNC(=O)C=Cc2cnc[nH]2)C(C)(C)C1 c12cccc(c1OC)NC2=O.C(=O)(C(C)(C)CF)NC1C(CNC(COC)=O)C1.CC C(=O)(CCCC(C)C)NC1CCC(Nc2ccc(OC)cc2)C1 c1(OC)nc(Cl)c(C(=O)NC2CC(CNC(C3(Cl)CC3)=O)C2(C)C)s1 CC1=C(CNC(c2cccc(C3CC3)c2)=O)CCC1 C(C(C(=O)NCC(O)C1(Cl)CC1)n1cc(-c2ccnn2C)nn1)OCCOC C12(CNC(c3ccn(COC)n3)=O)CCC(C1)N(C(C1(C)CCCO1)=O)C2 c1(C(CO)NC(C2CC2CO)=O)ccsc1 C(=O)(C(C)(C)CC(C)(C)C)N1CCC(NC(C=C(C)Cl)=O)CC1C1CC1 C=CCC(CC=C)C(=O)N1CCCC(CCO)CC1.C1(CCCOC)C(=O)N1 CS(=O)(=O)CCC(=O)NCCCOCCC(N1CC2C(C(N)=O)C2C1)=O C(=O)(C(C)C(F)(F)F)NCC(CC)NC(c1c[nH]nc1C1CC1)=O N1(CCC(=O)NCC(C)N(C)C(C2CCCCN2C)=O)CCCCCC1 CCC(CC(F)F)C(=O)N1CC2(CC2)CC1CNC(c1cnc2c(c1)CCC2)=O C(C(C(=O)NC(C)CCc1cn[nH]c1)NC(C1CC(C)=NO1)=O)SCC c1(N2C(CN(C(=O)C(O)CC(C)(C)C)C)CCC2)nc2ncc(Cl)cc2o1 N#CC(CC1CCCCC1)C(=O)NCCN(C(c1ccnnc1S)=O)C1CC1 CC12CC(C(=O)NCC(C3CC3)NC(=O)CC3CCCO3)(CCO1)C2 C=CCC(C)(C)CC(=O)NCC1(C(C)(C)O)CN(C(=O)CC2CCOC2)C1 c1(CC(=O)NCC(CN(C(=O)CC(C2CC2)C2CC2)CC)(C)C)ccnc(C)n1 C(CCCCC(=O)N1CCCCC(CNC(=O)CO)C1)SC c1(C(=O)NCC23CC(C)C2C3)cccc2nncn12.N12C3CCC1(CC3)C2=O c1(C(C)C)cccc(C(N2CC(O)(CNC(=O)C=Cc3cocn3)C2)=O)n1 C(=O)(C(C(C)C)NC(c1cccn1C)=O)NC(CC)C(C)C C1(CC)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)CCN1C(=O)C(C)=C1CCC1 Cc1nc(CC2CC2)sc1C(N1CC(C(C)NC(c2cnc(S)n2C)=O)C1)=O C1(OC)CC(CNC(=O)C(C)(F)F)N(C(=O)CN2CC(=O)NC2=O)C1 C(=O)(CC(O)C(C)C)NCC(C)C(=O)NCC1CCC2(CC2)C1 C1(CCC(N2CCC(n3cc(-c4ncoc4C(=O)O)nn3)C2)=O)NC(=O)NC1=O C1(C)(C(N2C(CN(C(CC3C(C)OCC3)=O)C)CCC2)=O)CC2(CCC2)C1 C(C)(C(=O)NCC(C)N(C(=O)CN1CCC(=O)NC1=O)C)(C(C)C)NC(C)=O Cc1cc(C(N2CCC(n3cc(CNC(=O)CSC4CC4)nn3)C2)=O)nnc1C c1(C(=O)NCC(CC)(CC)Nc2ncc(C#N)cc2F)cn(C)c(C)cc1=O c1(C(=O)NCC2N(C(C(CCC#C)O)=O)CCC(C)C2)ccc([N+](=O)[O-])c(C)n1 CC1C(NC(=O)Cc2csc(-c3ccoc3)n2)CCN1C(C1CCCOC1)=O c1(-c2cncc(CC(=O)NCCNCCO)n2)ccc2ccnc(O)c2c1 N1(C(COCCSC)=O)CCC(CN(C(C2CCSCC2)=O)C2CC2)C1 N1(C(Cn2c(C)ncc2)=O)CCC(CNC(=O)C(O)C2CCC2)C1(C)C N1(C(C2C3(CC(OC)C3)C2)=O)CCC(C(C)CO)CC1.C12(CCCC1O)CO2 CCCCCC(O)CC(=O)NCC(C)(C)NC(=O)Cc1ccccc1C(F)(F)F N1(C(c2cnc(NC)nc2)=O)CC2CCC(CNC(c3ncc(F)cn3)=O)C2C1 C(=O)(CS(=O)(=O)N(C)C)NC(C1CCCCC1)C(C)NC(=O)CCN1CCC1 N1(C(c2nc(=N)[nH]cc2)=O)CCN(C(c2nocc2Cl)=O)C2CC12 O=C1CC(CC(N2CCC(NC(=O)CCc3cnco3)C(F)C2)=O)CCCN1 C1(CNC(c2[nH]nnc2C2CC2)=O)(NC(C2CC=CC2)=O)CCC(F)(F)CC1 Cc1cc(C=CC(N2CCC(C)CC2CNC(C2CCOC2)=O)=O)c[nH]c1=N c1(C(N2C(CNC(CCc3cncc(C)c3)=O)CC2)=O)ccc2nncn2c1 c1(C(=O)NCC2CCCN2c2nccc(CO)n2)c(Cl)cc(Cl)cc1Br C(C(CC(F)(F)F)NC(CS(=O)(=O)NC(=O)C(O)CCSC)=O)OCC c1(NCC(=C)Br)nccc(=NCCCCCC2CC2)[nH]1 c1(-c2c(CC)non2)nc(-c2ccc(SC)cc2)nn1CCOC(C)(C)C C1(NC(CC2(OC)CC2)=O)CCCC(CCNC(c2cncc(Cl)c2)=O)C1 c1(CC(=O)C(C2(N)CSC2)=O)c[nH]ccc1=O.CCC(CC)=CCOC(C)=O N1(C(CC(CCCC)NC(=O)CC=C(Cl)Cl)=O)CCCN2CCCC2C1 Cc1nc(CCCC(=O)N(C)CC2CCCN2C(=O)C(C)c2ccsn2)cs1 C#CC1CN(C(=O)C(n2ccc(C)n2)C)CCN1C(=O)C(CC1CC1)OC C(=O)(C(CC1CC1)NC(c1ocnc1C(C)C)=O)N(CCCC)C N1(C(C(C=C)C)=O)CCN(C(=O)CCC(C)OC)C(c2ncc[nH]2)C1 C1(C)(NC(C(C)OC)=O)CCCN(C(=O)CCc2ccc(C)s2)C1 c1(C(N2CC(NC(C(CC)(C)O)=O)C(C(F)F)C2)=O)cnc2c(c1)CNC2=O c1(C(=O)NCC(O)CNC(C2(F)C3CCCC23)=O)ccc2sccc2c1 N1(C(c2c(COC)n(C)nc2)=O)CCOC2(CCN(C(C3CC3C)=O)CC2)C1 CC1(NC(C2CC(=O)OC2(C)C)=O)CCCN(C(=O)CCN2CCCCC2=O)C1 C1(NC(c2n(C)ccc2)=O)CCCCN(C(=O)CC2SC(=N)NC2=O)CC1 c1(C(N2CCC(CNC(=O)Cc3cccnc3)C23CC3)=O)cnc2cc[nH]c2c1 c1(NC(C2CCCN(C(C(C)C3CC3)=O)CC2)=O)ccc2c(c1)CCO2 c1(SC)nc(O)nc(C)c1C(N1CCC(O)(CN(C)C(c2cnsc2)=O)CC1)=O C(C(C(=O)NC1CCC1COC(C)(C)C)NC(C)=O)OC.C(=O)(C1=CCC1)NC c1(C(=O)OCC)noc2c1CN(Cc1cnc(C(C)(C)C)nc1)CC2 c1(C(N2CCC(NC(=O)CO)C(O)C2)=O)c(F)cc(Cl)cc1Cl N1(C(C2(F)C(C)C2)=O)CCC(CO)(NC(=O)CCCc2cnn[nH]2)C1 Cc1cc(C(=O)NC2C=CC(CC(=O)NCc3ncnn3C(C)C)C2)cc(O)c1 N1(C(C2C(C)C2)=O)CC2(CC2)CC1CNC(C1CC(N(C)C)C1)=O N1(C(C23CC(NC(CC4C(C)CCC4)=O)(C2)C3)=O)CCC(C(C)C#N)CC1 Cc1cccc2c(C(=O)NC3CCN(C(=O)Cc4cccc(F)c4)CC3)c[nH]c12 CC1(C)CC(C)(CNC(=O)C(F)CC2CCC2)CN1C(c1c[nH]cc(Cl)c1=O)=O Cc1nn(C)nc1C(=O)NCCOC1CCN(C(=O)C(c2c(C)n[nH]c2C)C)C1 c1(C(N2CC(C)(C(=O)NC(C3(O)CCCCC3)CC)C2)=O)ncncc1Cl C(=O)(C1=CC(C)(C)C1)N(C(CNC(c1ccnn1C)=O)C1CC1)C c1(SCC)cc(C)[nH]c(=NC(C)CCNC(=O)C=CCOC2CCOCC2)n1 CN1CCOC(C(N2CCC(C)(NC(c3cc(N)cc(O)n3)=O)C2)=O)C1=O C12(CNC(C(C3CCOCC3)OCC)=O)CC(CN1C(=O)Cc1cnsc1)C2 C(CC(C(C)(C)C)NC(=O)Cn1ncnn1)N(C(C(N1CCC(C)C1)=O)=O)C Cc1ccc(C(=O)NC2CCCN(C(C3CN(C4CCOC4)C3)=O)C2C)c(C)n1 O=C(C1=CC(O)CCC1)NCC1C2CC1N(C(=O)CSCc1cccc(Cl)c1)C2 N1(C(c2cc(C)c(Cl)cc2)=O)CC2(C1)CN(C(=O)C(C)O)CC(C)(C)O2 c1(C(=O)NC23CCCC2CN(C(=O)CCC2CCC2)C3)cc2cncn2c(O)n1 C1(CNC(c2c(NC)scn2)=O)CN(C(=O)CCC2CCN(C)CC2)CC12CC2 C1(C(=O)NCC(CNC(c2c(CC)cc[nH]2)=O)O)C2CCC(F)C12 c1(C(=O)NC2CC(C(N3CCCC(CC)C3)=O)OCC2)ccc(C#N)c(C)c1 CC1C(NC(=O)CC2C=CCCC2)CCCN1C(c1cnc(S)n1C)=O Cc1cc(C)c(C(N2CCCC(NC(C3C4(CC4)C34CC4)=O)C2C)=O)c(O)n1 N1(C(C=CC=COCC)=O)CCC(NC(=O)CC2CCOC(C)(C)C2)CC1C C1(C(=O)NCCn2cc(C(N(C(CC)C)C)=O)nn2)CC(F)C(=O)N1 O=C1CN(CCC2CC2)CCN1CC1CC=CCC1 C1(CC)(CC)CC(NC(=O)CSC(C)C)CN1C(c1cnncc1O)=O c1(C(N(CC(O)CNC(c2c(Cl)cnn2C)=O)C)=O)coc2c1CCCC2 N1(C(CC)=O)CCCC(C)C1CNC(C12CC(C1)C(C(=O)O)CO2)=O C(CC(C(C)(C)C)NC(C1CC(=O)CN1C(C1CC1(F)Cl)=O)=O)N(C)C N1(C(c2cn(C)c(=O)n2C)=O)CCCCCC(NC(C2CC23CCSCC3)=O)C1 CC1(NC(=O)CC2CCC(F)(F)C2)CCN(C(=O)C(=O)NCC(F)(F)F)C1 C1(NC(CS(CC)(=O)=O)=O)CN(C(=O)CCCNC(C)=O)C2CCCC12 C(=O)(C(F)(F)C(F)F)NC1C(C(=O)NC(c2ncc(F)cn2)C)COCC1 CC(C)C(CCN(C(=O)C(F)C1CCCC1)C)NC(c1ccc(Cl)[nH]1)=O c1(C(C(=O)N(CC(C)NC(COCCOCC#C)=O)C)(C)C)ccc(CC)cc1 c1(C(N(C(CNC(C2C(=C)C2)=O)C)C)=O)ccn(CCOC)n1 c1(C(=O)NC(C)C(=O)NCC(c2ccc(Br)s2)O)ccccc1C#N C(c1ccccc1F)=CC(=O)NC1(CNC(c2cc(C)c(C)o2)=O)CCCCC1 c1(C(N2CC(OCCNC(CC(C)(C)O)=O)C2)=O)cccc([N+](=O)[O-])c1Cl Nc1csnc1C(=O)NCC1CC(CNC(=O)C=C2CCOCC2)CO1 c1(C(N(C)CC2CC(F)CN2C(C2CCCN2C=O)=O)=O)cc2scc(Cl)c2[nH]1 C(=O)(CS(=O)(=O)NC(C)(C)C)NC(C)C(CO)NC(=O)CCc1cccnc1 C(C(C(=O)NCc1ncc(C)cc1C)C(C)(C)C)NC(C(C(CC)C)=O)=O Cc1nn2cccnc2c1C(N1CCN(C(=O)CCC2(C)CC2)C(C2CC2)C1)=O C(CCCCC(=O)NCC1N(C(C2CC2C#N)=O)CCC1(C)C)OCC N1(C(C2(OC)COC2)=O)CCC2C(C1)CN2C(=O)CC(c1ccccc1)N(C)C CC1CN(C(C2Cc3cscc3C2)=O)CC(C)CN1C(=O)C1=CS(=O)(=O)CCC1 C=CC1(C(N2CCOC(C(N)=O)C2)=O)CCN(C(c2cc(CC)oc2C)=O)C1 C(=O)(C(CC(C)C)NC1CCCCC1OC(F)(F)F)NCC(=O)OC C1(NC(Cc2c(C)con2)=O)CN(C(=O)CN(C)S(N)(=O)=O)CC1C N1(C(=O)CC2CC2C2CC2)CCC2CC12C(=O)N(C1CC1)CC1CC=CC1 Cn1ncc(Br)c1CN1CCCC(NC(C2(C)CNC(=O)C2)=O)C1 C(=O)(C(C)CCc1ccc(F)cc1)NCc1n(CCC)ncc1 CC(C(F)C(=O)NCC1CN(C)CCN1C(=O)Cc1cscn1)C(F)(F)F N1(C(c2[nH]n(C)c(=O)n2)=O)CC2(C1)C(NC(=O)Cc1cnccn1)CCS2(=O)=O N1(C(C2(C#N)C(C)C2)=O)CCC(O)(CNC(=O)Cc2cn(C3CC3)cn2)C1 C(=O)(C(C)C1=CCCC1)NC1(CC)CCN(C(C2(O)CCOC2)=O)CC1 Cc1c(C(N2CCCC(NC(=O)CC(C)CF)C2C)=O)[nH]c2ccc(Br)cc12 C(=O)(CCCCCC(C)C)NC1CCN(C(CCCCC(=O)NC)=O)CC1(C)C c1(C(=O)NCCNC2(C(F)F)CCNC2)ccc(N2CCCS2(=O)=O)cc1 C(C(F)(F)C(=O)N1CCN(C(C2(F)CCN(C(C)(C)C)C2)=O)CC1)OC c1(C(N2C(CNC(C(C)OC)=O)CC(F)(F)C2)=O)ccc2c(O)nc(S)nc2c1 CCC1=C(C(=O)N2CC(C3(NC(=O)C(F)CC4CCC4)CC3)C2)CCCO1 O=C(C1CC(O)c2ccccc21)N1CCC(n2cc(COCCO)nn2)C1 N(C1CCc2cccnc21)C(C1N(C(c2cc(C)c(F)cc2)=O)CCC(O)C1)=O C=CCCCCCCC(=O)N1CC(F)CC1CNC(=O)CC1CCOC1=O c1(N(C)C)ccc(C(N2CC3C(C2)N3C(c2ccc[n+]([O-])c2)=O)=O)cc1F C1(CC(=O)NCC2C(NC(CCOCC#C)=O)C2)CCC(C)(C)CC1 C(=O)(C(F)C(C)C)NC1(COC)CN(C(=O)CCC2CCC(=O)NC2)C1 N1(C(c2c(C)nn(CCO)c2)=O)CCN(C(=O)C(C)(O)C2CC2)C2(CC2)C1 C(=O)(C(C(C)(C)C)N1CCCC1=O)NC(CC)(C)CNC(=O)CCCC1CCC1 C1(CNC(C2(C)CCC(C)C2)=O)CN(C(=O)CC2CCC(C)(C)CO2)CCCO1 C1(CC)(CO)CCCN(C(=O)COC2CC(NC(C3CCCC(C)(C)C3)=O)C2)C1 C1(CNC(C(C)(C)c2cnco2)=O)CN(C(=O)C2=CSCS2)CCO1 C1(C(=O)OC)CCC(C(=O)N(CC(C)(C)CNC(C2COC(=O)O2)=O)C)CC1 C=CC1(C(N2CC(C)(C(=O)OC)C2)=O)CCN(C(=O)CC2C=NN(C)C2=O)C1 C(CC(F)F)(C(=O)NC1CCS(=O)CC1)NC(CC1CC(CC)C1)=O C=CC1CN(C(=O)Cc2ccc(N(C)C)cc2)CC1NC(c1ccc(CO)o1)=O c1(CN2C(C(N3CCC(CCO)CC3)=O)CNCC2)cc(O)c(O)cc1O CC(C)(C)C1=NOC(C(=O)NCCCNC(=O)CNC(c2ccco2)=O)C1 n1(CCOC)ccc(C(=O)NCC2CCN2C(=O)Cn2ccnc2C(C)C)n1 C=CCCCCCCC(=O)NC1CCC(NC(c2nnn(CC)c2C)=O)CC1 c1(C(=O)NCC(CC)NC(C(CCC)OCC)=O)cc2cccc(C)n2n1 c1(C(=O)NC)cc(=NC2COc3c(Cl)cccc32)cc[nH]1 C12C3CC1N(C3)C2=O.c1(C(C)=O)ccc(C(C)O)cc1.c12cn(nn1)CC(=O)N2 Cc1c(C(N2CCCN(C(C3C4CCC(F)(F)C34)=O)CC2)=O)cccc1O C1(C(=O)NCc2c(CC)nns2)CCC2(CC2)N1C(C1COCC(C)O1)=O N1(C(C2CCC(OC)CC2)C(=O)NC2CC2)Cc2cccc(C)c2CC1C(=O)O CCC(C)C(O)C(=O)N(CCNC(c1cc(C2CCCCC2)n(C)n1)=O)CC.C(C)O O=C(N=c1cc2n([nH]1)CCCC2)C1N(C(C2CCC2)=O)CC12CCCC2 C(=O)(CCCC(=O)N1CCC(NC(=O)CC2CCC3CC3C2)C(C)C1)OC C=C(C)CC(C)C(=O)NCC(C1CCN(C(C2(n3cccn3)CC2)=O)CC1)C Cc1ccc(C)c(C(c2ccccc2)NS(=O)(=O)Cc2cc(C)no2)c1 CCCCC(C)CCC(=O)N1CCC(C)(NC(c2ccc(C(F)(F)F)nn2)=O)C1 Cc1cc(C)c(C(=O)NCc2ccoc2C(=O)NC(C2CC2)C2CC2)cn1 C1(OC)CN(C(C2CCC(C(F)(F)F)CC2)=O)CC1NC(c1occ(C)c1C)=O c1(C(N(CCC(C)NC(=O)CC(C)F)C)=O)cn2cccnc2n1 c1(C(=O)NC2CC2CNC(C2CCCC2)=O)csc(-c2cccs2)n1 CC1CC2(CCN(C(c3ccnc(O)c3)=O)CC2)CN1C(C1CC1(F)F)=O O=C(CN1C(=O)Cc2cc(F)ccc21)NCC1CC1CNC(C1C2CCCC12)=O Cc1cc(F)c([N+](=O)[O-])cc1C(=O)NC1CN(C)CC1(F)F N1(C(C(C)CN2CCOCC2)=O)CCCN(C(=O)CCCC(F)(F)F)C(CO)C1 C(CCCCC(=O)NC(C)C(C)NC(c1cncc(C)n1)=O)NC(C)=O c1(OCCCC)ccc(CCCNC(=O)Nc2csc(CCN)n2)cc1 N1(C(C(CC(C)C)N(C)C)=O)CCC(C(N2CCOCC(C(C)C)C2)=O)C12CCC2 Cn1cc(CNC(C2N(CC3(NC(N)=O)CCCC3)CCC2)=O)c2cccnc12 CCC(C)(CC)C(=O)NC1(C(=O)Nc2ccc(NS(C)(=O)=O)cc2)CCOC1 N1(C(Cn2c(C)nnn2)=O)CC2(CCC(CNC(C3(C(C)C)CCCO3)=O)O2)C1 c1(CC(=O)NC(N)=O)cc(F)cc2c1OCOC2.C1C(C)(C)C(=O)N1C C(CC(C(=O)NCCCSCC)NC(c1cccc(CO)c1)=O)=CC N(S(=O)(=O)N1CC(O)C1)(C(C)C)C1CC1 c1(CNC(C(CCNC(=O)CC2CC(=O)NC2=O)O)=O)cc(F)cc(F)c1 C(=O)(CC(O)C(C)CC)NC1CCC(CCC(=O)NC(C2CCCC2)CC)C1 c1(C(N(CC(C)NC(Cn2c(C(C)C)ncc2)=O)C)=O)c(Br)nnn1C C1(CNC(c2cnc(OCC)s2)=O)C(C2CC2)CCN1C(=O)COCCF N(C1CCCc2c(O)cccc21)Cc1cccc(S(C)(=N)=O)c1 c1(CC(N2CCC(c3cccc(Cl)c3)(NC(C)=O)C2)=O)cc(O)nc(O)n1 c1(CC(N2C(CCNC(c3cc(C4CC4)on3)=O)CCC2)=O)ccc(Cl)cc1F C1(C(N2CC(C)C(NC(c3ccc(C(F)F)s3)=O)C2)=O)CC2CCC1CC2 c1(C(=O)NC(CN(C(=O)Cn2nccc2C)CC)C)ccc(P(C)(C)=O)nc1 C1(O)(CNC(COc2cc(C)on2)=O)CCN(C(C2(O)CC2)=O)C1 c1(CC)ccnc(C(=O)NCC2COC(CNC(=O)CSc3nncs3)C2)c1 C(CC(=O)N1CCS(=O)(=O)CCN1)N1CCC(C(C)=O)CC1 c1(C(=O)NC2(C)N(C(c3cncc(OCC)c3)=O)CC2)cc(F)c(OC)c(Br)c1 c1(NCC=CC)ccc(S(=O)(=O)N2CCCC(C(C)C)C2)cc1Br c1(C(CNC(C2CC(C(C)(C)C)C2)=O)O)ccc(F)cc1Br CCC(C)C(CNC(=O)CN(C(c1ccc[n+]([O-])c1)=O)CC1CC1)CO O=C1CCC(COC(c2cn(C3C=CCCC3)nn2)=O)O1 C1(C(=O)NC(C)C(C)(C)NC(c2cccc(-n3cncn3)c2)=O)COCCOC1 C1(CNC(C=CC(CC)C)=O)COCCN(C(c2cc(C(C)C)[nH]n2)=O)C1 Cc1ccc2occ(CNC(C34CC3CN(C(=O)CC35CCCC3C5)C4)=O)c2c1 c1(CC(=O)NC2CCC(CCNC(C3(CC(C)C)CC3)=O)C2)ccc(OC)cn1 C1(NC(C2(COC)CCCO2)=O)CCCCN(C(c2ccc3c(c2)CC3)=O)C1 c1(OC)c(F)cc(F)c(N2CC(OCCNC(=O)C(O)C(C)C)C2)c1[N+](=O)[O-] CC1=CCC(C(N2CC=CC(NC(=O)C=CCn3cncn3)C2)=O)CC1 N1(C(c2c(OC)ccs2)=O)CC2COCCC2(NC(c2ccn(C(F)F)n2)=O)C1 C(CCCCC(C(=O)NCc1nnn(C)n1)N1CCN2CCCCC2C1)OC C1(CCCC)CN(C(c2nn(C)cc2Cl)=O)CCN1C(=O)C(n1cc(Cl)cn1)C N1(C(C(C2CC2)OC)=O)CCCC2(CCN(C(c3ccn(C(C)(C)C)n3)=O)C2)C1 CC1CN(C(=O)CC#N)CC(C)N1C(=O)CCCc1ncco1 CCCCCCCC(=O)N1CCC(NC(c2cc(Br)cnc2N)=O)C1 Cc1ccnn1C=CC(=O)NC(CCCNC(=O)C=CC(C)C)c1ccccc1 c1(CC)ccc(CC(=O)NCCCCCCN(C(=O)C=CC(C)CC)C)cc1 c1(C(=O)OCC=CC2(C)COC2)ccnc(CO)c1 c1(C(=O)NC(C2(O)CN(C(c3c(Cl)cncc3Cl)=O)C2)C)cccc(S(C)=O)c1 CC(C)(C(=O)NCCCNC(=O)C1=CC2CC=CCC12)C1=CCSCC1 C1(NC(c2cn(C)nc2)=O)CN(c2ncc3c(ncn3C)n2)Cc2nccn2C1 S(=O)(=O)(c1cccc(N2CCNCC2)c1)Nc1ccc(OCC(C)C)c(F)c1 Cc1ccn(C)c1C(=O)NCC#CC(=O)NCC(C)S(N)(=O)=O N1(c2nc(C(C)C)nc(N3CCC(C#N)C3)c2)CCn2ncc(Br)c2C1 c1(NCC23CC(NC(C(C=C)O)=O)(C2)C3)cc(Cl)ncn1 N1(C(CNC(CCC)=O)=O)CCCC2(CCN(C(C3OCCO3)=O)C2)C1 C1(NC(CN(C)CC)=O)CN(C(c2ccc(F)c(O)c2F)=O)C2(CCCC2)C1 N1(C(=O)OCC)CCN(C(=O)NC2CCCOC2c2ccccc2)CC1 N1(C(CCN(CC)CC)=O)CC(NC(=O)Cc2sc(O)nc2O)CC12CCOC2 CCCC(C(=O)N(CC(=O)NCc1ccccc1F)C1CC1)NC(C)=O c1(OC)cccc(C(C(=O)NCC2CC2NC(c2cnc(C)o2)=O)C(C)C)c1 C(=O)(CC(C)CC(C)(C)C)N1C(C)CN(Cc2nc(-c3ccccc3)cs2)CC1 Cc1cc(C(=O)NCC(F)CNC(=O)CC2CC(C(F)F)C2)no1 C1(NC(=O)N(CC=CCCOC)C2CC2)CCN(C(=O)C(C)(C)C)C(C)(C)C1 c1(C(=O)NCC2C(NC(c3[nH]cc(C#N)c3)=O)CC2)onc2ccccc12 N(C(=NC(C)C=C)N1CCc2cc(Br)sc2C1)C(CC#C)C(=O)OC N1(C(C2(C)CCN(C(c3cc(O)cc(O)c3)=O)C2)=O)C2CCCC1COC2 C1(NC(C2C(OCC)C2C)=O)COCCC1NC(c1[nH]c(=N)sc1C(F)(F)F)=O CC1(C)CC(O)CN1C(=O)C(=O)OC1CN(C(=O)COC(=O)Nc2ccccc2)C1 C1(C)(COC)CN(C(c2ccc(SCn3cc(C4CCCC4)nn3)o2)=O)C1 C1(CC(=O)NCC2(NC(c3c(Cl)cn(CC)n3)=O)CC2)CC(=O)NC(=O)C1 C1(CN(C)C(C2(C)CC2(F)F)=O)CCN(C(=O)CN(C)C2CC2)C1 c1(OC)cnc(C(F)(F)F)cc1C(N1CC(O)CC1(C)C1CC1)=O C(=O)(C1=C(C)OCCC1)N(C1CCC1)CC1C(CCC)CCC1.C1C(=O)N1 N1(C(c2c(C)n(C)cn2)=O)CC2CC1CN2C(C1CC1C(C)(F)F)=O c1(OC(C)=O)ccc2c(c1)NC(=O)C2(C)CO.C(C)(C)(C)OC(=O)N(C(C)=O)C1CC1 c1(C)cccc(O)c1F.c1(NC(=O)OC(C)(C)C)conc1CONC=O C1(CCC(=O)NCCCC(C)NC(=O)CN2CC3CC3C2)CCCCN1C c1(C(=O)NCC2(C(F)F)CCN(C(C3C(C)(C)C3)=O)C2)cc2c(Cl)ccnc2s1 C1(CNC(c2c(CC)cno2)=O)CCCN(C(=O)Cn2cnc([N+](=O)[O-])c2)CC1 C12(CN(CCO)C(C3(c4ccc(F)cc4)CC3)=O)CC1CN(CC1(C)CCC1)C2 C1(NC(COC2CN(C(C)=O)C2)=O)COC2(C1)CN(C(C1CCCC(O)C1)=O)C2 c1(C(N2C(C(C)(C)CNC(C3CCCO3)=O)CCCC2)=O)cnc2n1CCOC2 N1(C(CCOCCC)=O)CCCN(C(=O)CC2CC(C3CC3)C2)CC1C c1(C2N(C3CCN(C(CSC4OCC(C)C4)=O)CC3)CCC2)ccc(=O)n(C)c1 Cc1cccc2c1OCC2C(=O)N1CCC(CNC(c2nc(C)n(C)n2)=O)CC1 C1(C(N2CCC(COCC)C2)=O)CC12CC(NC(=O)C=C1CCOCC1)C2 CCCCC(C(=O)NCc1cc(C)c(C(=O)NCCC(C)(C)F)o1)N(C)C C(=O)(CCC#Cc1ccccc1)NC(C1(O)CN(C(C2CC2(F)F)=O)C1)C N1(C(Cc2c(C)ncnc2)=O)CCC(C2CC2)C1CNC(=O)C=CC(F)(F)F N1(C(=O)Cc2ccns2)CC2CCCC(C1)N2Cc1cnon1 C1(NC(CC2(OC)CC2)=O)CC2CC1CC2C(=O)N(C(C)C(F)F)CCO c1(C(C)=O)cc(CCC(=O)NC2COCC2NC(=O)C(=O)NC2CC2)oc1C c1(C(N(CCCCN(C(C(CC#C)C2CC2)=O)C)C)=O)ccc([N+](=O)[O-])s1 c1(C(N2CCCC(C)C2CNC(=O)CC2CC=CC2)=O)ccnc2c1nnn2C C1(CC(=O)OCC)CC(N=c2ccnc(N3CC(OC(C)C)C(F)C3)[nH]2)C1 N1(C(C2CCCCC2O)=O)CCC2CN(C(C3CC(O)C3)=O)CC2C1 C1(c2ccccc2)(C(N2CCC(OC3CCOCC3)C2)=O)CC2(CC2)C1 C(CC(CC)C(=O)NC12CC(C1)N(C(=O)CCC1CCCN1C)C2)=CC c1(C(N2CCC(O)(C(C)NC(C(C)C)=O)C2)=O)cnn(CC(C)C)c1C1CC1 C1(CNC(C(C)(C2CC2)OC)=O)CCC2CN(C(=O)Cc3ccns3)CCC2C1 N1(C(CCCOCC)=O)CCN(C(=O)COCc2ccccc2)CC(O)C1 C1(NC(CC(=O)OC)=O)CCN(CCNC(C2CCCC2C(C)C)=O)CC1 c1(C(N(C(CNC(C2CC2C(F)F)=O)C2CC2)C)=O)cccc(Br)c1 C1(NC(C(CNC(c2ccccc2Cl)=O)O)=O)C2CCC3C(C2)CC13 Cc1oc(C(C)C)cc1C(N1CCC(O)(CN(C)C(C2CCCC(O)C2)=O)C1)=O c1(OC)ccc(C)cc1NC(=O)CSc1nnc(SC)n1C1CCCC1 CC(C(C)(C)C(=O)N1C2CSCC1C2)NC(=O)CCCC1CCCO1 CCC(CC)C(C)C(=O)NC(C)C(=O)NC(C(N)=O)C(C)CC c1(C(=O)NC(C2N(C(C(C)OCC)=O)CCC2)(C)C)cccc(OC(F)(F)F)c1 Cc1cc(C(=O)NC2CCOC(CNC(=O)CSc3nc[nH]n3)C2)cc(C)n1 N1(c2n(CCC#C)c(-c3cccc(Cl)c3C)nn2)CC2(C1)OC(=O)NC2C c1(C(=O)NCCN(C(=O)CC2CC23CC3)C(C)C)ccc(C(=O)N)o1.C1(CSC)CC1 CCC(CCCC(=O)N1CC(n2cnnc2)C1)NC(c1cnc2n1CCC2)=O N1(C(CCSCC)=O)CC(F)(F)CC1CCNC(C1CCC(C(F)(F)F)CC1)=O C1(O)(COC(CNC(CCOCCC)=O)=O)CCCN(C(=O)C(C)C)CC1 N1(C(c2c(OC)ccs2)=O)CCC(NC(C2(OC)CCCC2)=O)C2(CCC2)C1 N1(C(c2cc(C)sn2)=O)CCCCC(C2CN(C(C3C4CCC(=O)C34)=O)C2)C1 c1(SC)ncc(C(=O)N(CC(C)N(C)C(c2oncc2C)=O)C)s1 c1(C(=O)NCC2C=CC(NC(c3c(C)ncnc3)=O)C2)ccc(OC(F)F)c(F)c1 C1(NC(c2c(OC)cc(C)s2)=O)C(C)CCN(C(c2csc(C)c2)=O)C1C S(=O)(=O)(c1ccc(C(=O)NC2CC(NC(=O)COCC(F)F)CC2O)s1)N(C)C C1(F)(C(N2C(CNC(C(C)(C)n3cnnn3)=O)CC2)=O)CC=CCC1 N1(C(C)C)CC(C(=O)NCC(CNC(c2ccccc2C(F)F)=O)CO)CC1=O c1(O)ccc(C)cc1C.c1(Cc2cc(C)no2)nc(C)nn1-c1nccn1C c1(C(N2CCC(CCNC(C3CSCCS3)=O)C2)=O)cnn2c1S(=O)(=O)NCC2 N1(CCCCCNC(CSC)C)CCN(C(=O)C(C)(C)n2ccc(C)n2)CC1 C(=O)(C1CC(=O)c2ccccc21)N(CCN(C(C1=NOC(C)C1)=O)C)C N1(C(CCC(=O)OCC)=O)CCC(C)(C)C(NC(=O)Cc2c[nH]nc2C)C1 C1(C(N2CC(CNC(=O)C(=O)NCc3c[nH]cc3C3CC3)C2)=O)CCCCC1 C(=O)(CC(C)(C)N(C)C)N(CC(C)OC)CC1CC1.C(=O)(CCCC1CC1)NC CC1(F)CN(C(C2(C)CCCO2)=O)CCN(c2ncc(Cl)c(O)n2)C1 C1(C(=O)NCCOCCNC(c2c(C)nc(C)o2)=O)COc2ccc(F)cc2C1 n1(C(C(C)C)(C)C)cnc2c(N3CCCC(F)(F)C3)ncnc12 c1(OCc2c(F)ncc(OC)c2)nc2ccccc2nc1N1CCC(C)=C(Br)C1 Cc1c(C2CCCN2C(=O)C(=O)NC2(C)CCCOC2)cccc1Br CCC(C)(C)CCCC(=O)N1CCN(CC(=O)NCC2(C)COCCO2)CC1 C1(C(C(=O)OC)NC(=O)CC2CCNC2=O)CCCCC1 c1(C(N2CCC(C(C)(C)NC(c3cccs3)=O)CC2)=O)ccc(F)c(Cl)c1 N1(C(C2CCC(C(N)=O)O2)=O)CCOCC(CNC(c2n[nH]cc2F)=O)C1 N1(C(C2N(C(CCC)=O)CSC2)=O)CC2CC(NC(=O)C(C)C(C)(C)C)CC1C2 N1(CCC(CCC(=O)NCC2CC2)O)CCCCC1=O Cc1cccc2c1CC(C(=O)NCCCCNC(=O)N)NC2.c1(O)ccccc1F N1(C(C=CC(=O)OCCCC)=O)CC2C(CNC(=O)C(c3cncnc3)C)C2C1 c1(C(N2CC(NC(=O)C=CCn3cncn3)C(F)C2)=O)cc(F)cnc1O c1(C(N(CCC(C(C)(C)C)NC(=O)OC(C)(C)C)C)=O)nc2cc(Br)ccc2o1 CC(C)CC(CNC(=O)C=Cc1ccco1)C(=O)N1CCn2cnnc2C1 c1(NC(=O)NC(CC)C(F)(F)F)cc(C(C)(C)C)ccc1OC c1(C(=O)NCCNC(c2n(C=C)nnc2)=O)cc2ccccc2cc1N c1(CNC(C(C)N(C)CC2CCCCN2C(C2CC2)=O)=O)ccc(Cl)cc1Cl N1(CCCNC(=O)CCn2cncn2)CCN(C(c2cc(F)c[nH]2)=O)CC1 Cc1ncc(CCC(N2CCC(N(C(=O)Cc3cc[nH]c3)C)C2)=O)o1 N1(C(C(c2ccc(Cl)c(Cl)c2)C)=O)CCCC(CO)(NC(c2nc(O)n[nH]2)=O)C1 C1(CNC(C(C)N(C)C)=O)CC2CCC(C1)N2C(=O)CC1Cc2ccccc2O1 N1(C(C2(NC(C)=O)CCCC2)=O)CCCC2CN(c3nnc(CO)s3)CCC12 c1(C(=O)NC(C2CCN(C(C(C)(C)OCC)=O)C2)C)cnc(S)nc1 c1(CCC)nn(C)c(C(N)=O)c1NC(C12CC1CN(Cc1ccnc(C)c1)C2)=O Cc1nc(NCCCN2CCC3CC3C2)cc(=NCC(F)(F)CC2CC2)[nH]1 c1(C(=O)CSc2c(F)cc(F)cc2F)ccc2sccc2c1 CCC(CC(F)(F)F)NC(=O)CC1COCCN1C(=O)C(c1cccn1C)=O O=S(=O)(c1ccc(OC(F)F)c(F)c1)NC1CCc2nccn2CC1 C(=O)(CCC(F)(F)F)N1CCC(C(C(=O)NC2(CO)CC3CCCC23)F)CC1 c1(NC(N2CC(CNC(C)=O)OCC2)=O)ccc(Br)c(N(C)C)c1 Cc1cc(OCC(=O)NCCC2(NC(C3CC3C3CC3)=O)CC2)cc(C)c1 C1(NC(C(=O)NCC2CC2)=O)CN(C(c2ccc3nc[nH]c3c2)=O)CC2(CC2)C1 c1(NC(C2N(C(c3n(C)ncc3)=O)C3CCC2C3)=O)n[nH]c2cc(Cl)ncc12 C1(C(=O)NC2CC(NCc3cc(Cl)cc(C)c3O)C2)CCc2nnc(O)n2C1 c1(C(N(CC(CNC(c2cccc(OC)c2Cl)=O)O)C)=O)c(C)cc(F)cc1C C1(OC)CNC(C)(CNC(C2COCC2n2ccnn2)=O)C1 C12(C(N(CCCOCCNC(c3ccoc3C(N)=O)=O)C)=O)CCCC1CC2 c1(N2CC3C(CO)(C3)C2)nc2c(c(=NCC(=O)N3CCCCCC3)[nH]1)COC2 c1(C(=O)NC2CCCN(C(CS(=O)(=O)NC)=O)C2)c(C)nc2sc(C)cn12 CC1CN(C(=O)C=C(Cl)Cl)C(C)CN1C(=O)CN(C)C C(=O)(C#CC1(CC)COC1)NC(CC=CC)C(=O)NC(C)COC CC(CC(F)F)C(=O)NC1CCC(CNC(C2CCOC2C2CC2)=O)CC1 C1(C)(C(N2CCC(NC(COCCCCCC)=O)C2)=O)CC(C)=NO1 N1(C(C(COC)C)=O)CCCCC12CN(C(=O)C(C)c1cncs1)C2 N1(C(NOCC(=C)C)=O)CCCCC1Cc1ccccc1 C(C(CC(C)C)C(=O)NCCCN(C(=O)C(C)CSC)C)NC(CC)=O C1(CN2C(c3c(S(C)(=N)=O)c[nH]n3)CCC2)CCCC2(CNC2)O1 n1(CCN(C(=O)CN2CCCC2c2ccc(C)cc2)CC)cnc2ccccc12 C(=O)(N(CCC(=O)N1CC2(CCNC2=O)C1)OC)c1c(CC)[nH]cc1 C1(NC(C(CC)(C)CC)=O)CN(C(c2cc(C)cc(C)c2O)=O)C2CCCCC12 C(=O)(CC1c2ccccc2Oc2ccccc21)Nc1c(C(CC)C(N)=O)nco1 N1(C(c2cc(C)ncc2C)=O)CCC2CN(C(c3occc3C3CC3)=O)CCC12 C1(=CC(=O)NCCCN(C(C)C)C(C2(CCNC(N)=O)CC2)=O)CCCCC1 C1(CCNC(CN(C)C(C2COCOC2)=O)=O)CCCCC1O CCCC(CC)S(=O)(=O)N(C(c1ccc(Br)cc1)C(C)C)C c1(C(N(C2CN(C(C(CC)O)=O)C2)C)=O)csc(C)c1C C(c1cccc(Cl)c1Cl)=CC(N1CC(O)(CNC(C2CCC(=O)C2)=O)C1)=O n1(CC(=O)NC(C(C)(C)C)CNC(C2CC2C#N)=O)ccc(=O)c([N+](=O)[O-])c1 c1(CC(C(=O)OC)CNCC(O)C2CC2)ccc(Cl)cc1F c1(COC(C(=Cc2ccccn2)C)=O)ccc(F)cc1N C(c1cccnc1)=CC(=O)NCCC1CCCN(C(=O)CC2(CO)CC2)C1 C1(C(N2CCC(NC(c3ccc(Br)o3)=O)(CF)C2)=O)CCCC(F)(F)C1 CC(C)C(C)CC(=O)NCCc1ocnc1CNC(c1cscc1F)=O N1(CC(=O)NCC(C)OCCC(C)C)CCOC(COC)C1 N1(C(c2c(CC)noc2)=O)C2CCC1CN(C(=O)C#CC1(C)CCCO1)CC2 CCCCCCC(CC)C(=O)NC(C1(O)CCN(c2cc3nncn3cn2)C1)C C(=O)(CCCCCNC(=O)CNC(=O)CCC1CCCO1)OCC C(=O)(C(C)(C)CS(N)(=O)=O)NC(C)CC1CN(C(C2CN3CCN2CC3)=O)C1 c1(CC)cc(N(c2ccnc(N3CCSCC3)c2)CC)c(NC(c2cn[nH]c2)=O)cn1 C1(NC(=O)CCCCCF)CN(C(c2coc(Cl)n2)=O)CC2(CCC2)C1 c1(CNC2C(C)CN(C(c3cc(O)nc(O)n3)=O)C2)ccc2c(Cl)ccnc2c1 C(=O)(CCCn1cc(CC2(C)CCC2)nn1)NC1(COC(C)C)CC1 C1(CC)CN(C(c2cc(F)ncc2Br)=O)CCN1C(c1cnc[nH]1)=O C1(N(C(C2(C=C)CC2)=O)CCO)CCCN(C(=O)CN2CCCN(C)CC2)C1C CCCC(C)(CC)C(=O)NC1CCCN(C(=O)Cc2cnco2)CC1 CC1(C)C(N)C2CCCN(C(c3cc4cc(Br)cc(Cl)c4[nH]3)=O)C12 c1(C(=O)NC2C(CNC(CCC(C)SC)=O)COC2)ccc(N)c(Cl)c1 c1(C(N2CC(CC)N(C(c3oncc3C)=O)CC2)=O)nc2ccccc2o1 N1(C(C(C)(F)F)=O)CCOC2(CCN(C(=O)CNC(c3ccco3)=O)C2)C1 N1(C(=O)NC2CCC(COC)C2)CC2CCC1C(CNC(C)=O)C2 C1(CCNC(C(CC)C)=O)CCCN(C(=O)CC2CC3CCC2O3)C1 N1(C(C2CCC(C)CC2)=O)CCC2(CCOCC2)C(CNC(C2(O)COC2)=O)C1 Cc1cc2nccnc2cc1C(=O)NCCC(C)NC(C1CCC(F)(F)C1)=O C1(NC(c2c(C)nn[nH]2)=O)CCCCCC1NC(c1cnco1)=O Cc1ncc(Cl)c(C(=O)NC2CCN(C(=O)CCOCC3CCCO3)C23CC3)n1 N1(C(C2CCC(NC(C3CCN(C)C3)=O)CC2)=O)CCN2C(=O)NCC2C1 C1(OC2CCN(C(C(=O)N(C)C)=O)C2)CCN(C(=O)C=Cc2cocn2)CC1 Cn1nccc1NC(=O)CC1(NC(N2CCC(CC3CCC3)C2)=O)CC1 c1(C(=O)NC2CC(CNC(c3c(C)n(C)nc3)=O)C2)cc(Cl)cc2c1OCC2 C1(C(=O)NCC(C)CNC(=O)COCc2ccnc(O)c2)CCC(F)(F)C1 C#CCC(C)(CC)C(=O)NC(C)CNC(c1cc(N2CCCCC2)ccn1)=O c1(OC)ccc(CNc2ccc(C(=O)NCCC3CC3)nc2)c(Cl)c1Cl N=c1ccc(CC(N2CCCC2c2ccc(Br)s2)=O)n[nH]1 C(CCC(C)C)(C(=O)NCCN1CC=CCC1)NC(C(C)OCCCC)=O C(CN=c1[nH]c(=NCC(C)(C)CCC#N)[nH]c2c1CCCC2)N(C(C)C)C(C)C C(=O)(CCCCCCCCC1CC1)N(CC1C(NC(=O)Cn2cncn2)C1)CCO c1(C(=O)NCC2(CN(C)C(c3ccccc3F)=O)CC2)nccnc1C(N)=O C1(CNC(=O)CCC2CCOC2)CCCCN1C(=O)CCCc1cccc(Cl)c1 Cc1cc(C(=O)NCC(C(C)C)NC(C2CCCC2(C)C)=O)ccc1C(C)C N1(C(C(C)(F)F)=O)CC2CCC1CC2NC(c1c[nH]c2nccc-2c1)=O c1(OC)ccc(C(=O)NCC(C)N(C)C(C2CC2C(N)=O)=O)cc1Br CC(C)CCC(F)C(=O)NCC1CCCCC1C(=O)NCC1CC2CCC1O2 N1(C(C2CC(OCC#C)C2)C(=O)NCc2conc2C)CCCCC12CCC2 c1(C(N2CCC(C)C2c2cn(CCCN(C)C)nn2)=O)cc2n(n1)CCCO2 N1(C(c2cnn(CCCC)c2C)=O)CC(NC(c2coc(Cl)n2)=O)C2(CC2)C1 c1(C2(C(=O)NCC3C(NC(C4CN(C(N)=O)C4)=O)CC3)CC2)ccnc(Cl)c1 c1(C(=O)NC23CC(NC(CC=C(C)C)=O)(C2)C3)cc(C)ccc1C Cc1nc(C)c(CC(N2CC=CC2CNC(c2coc(Cl)n2)=O)=O)c(O)n1 c1(C(N2CCC(CNC(c3c(C)cns3)=O)C2)=O)ccc(C(C)(C)C)c(F)c1 C1(C(=O)NC2CN(CC(F)(F)F)C2)CCCN(C(=O)C=Cc2cnc[nH]2)C1 C(=O)(CC(C(F)F)NC(C1CC2(CC2)CO1)=O)NCCNC(COC)=O C1(C(N2C3CCC(NC(=O)C4=CCC4)(C3)C2)=O)Cc2ccccc2O1 C1(CC(=O)NC2C3CN(C(c4cc(-c5ccco5)[nH]n4)=O)CC23)CC2CCC1O2 N1(C(Cc2cn(CC(C)NC(=O)OC(C)(C)C)nn2)=O)CCC(C)C1C(C)(C)C C(=O)(C1=CC(C)(C)C1)N(C(C)CNC(=O)C(c1cccc(N)c1)O)C C12(C(=O)NCC(CC(=O)NC3CCCC(C)(C)C3)OC)CCN(CC1)CC2 N1(C(c2ccncc2F)=O)CCC2(C=C(C(=O)N3CCC(CF)CC3)C2)C1 c1(C(CO)N(C(=O)NCC(c2ncccn2)(F)F)CCO)cccc2ccccc12 c1(CC(=O)NCCCCCNC(=O)COC2CCOC2)cccc2ccsc12 C=CC(C)CC(=O)N1CC(c2ocnc2CNC(=O)C(C)CF)C1 C(=O)(CCC(C)(C)C#N)N1C(CNC(CCC2ON=C(C)C2)=O)CCCC1 CC1C(=O)NCCN1C(C1CN(Cc2ccc(N(C)C)cc2)C1)=O c1(C(=O)OC)nc(=NCc2nccs2)c(C#N)c[nH]1 C=Cc1ccc(C(N2CCCCC(CNC(C3C(C(F)F)C3(C)C)=O)C2)=O)cc1 C(CN=c1[nH]c(=NCC2CCOC2C)c2[nH]ccc2[nH]1)c1nc(C(C)C)sc1 c1(C(=O)NC(C2NCCOC2(C)C)(C)C)csc(Cl)c1Br C(C(CNC(=O)C(C)Cc1cnn(C)c1)C(F)(F)F)NC(CCC(=C)C)=O Cc1cc(F)c(Br)cc1C(=O)N(C1CN(C(c2ccccc2O)=O)C1)C c1(C(N2C(CNC(C3N(CC)CCCC3)=O)COCC2)=O)ccc(O)nc1Cl c1(C(=O)NC2(CC)CCCN(C(=O)CC3CC3)C2)ccc2c(c1)C(=O)NC2=O c1(C(=O)NCC2(OC)CN(C(C3(OC)CC3)=O)C2)cc(F)c(C)c(N)c1F c1(-n2cc(C(C(=O)NC)N(C)Cc3ccnn3C)nn2)ncc(C)cn1 C1(CNC(C2C=CCC2)=O)CC2CCCC(C1)N2C(=O)CCc1ccc(O)nn1 c1(SCC)cncc(N2CCC(C3CCC(=O)NC3)C2)n1 C(C(=O)NOCC=C(C)C)(C1CN(C(=O)C(C)n2cccc2)C1)OC C1(N(Cc2nnc(C)o2)CC)CC(NS(C)(=O)=O)C12CCC2 c1(NC(c2cccc(C(F)F)n2)=O)ccc(F)cn1 Cn1nnc2c1CC(C(=O)NC1CC1CNC(C1CCC3(CC1)CC3)=O)CC2 O=C(N=c1[nH]ncn1-c1ccccc1)NCc1ccccc1-c1ccc(F)cc1 C1(CNC(COCCC=C)=O)CCN(C(=O)C(c2ccc(Cl)c(F)c2)O)C(C)C1 c1(C(=O)NC2CN(C(CCCCCCCCC)=O)C(C)C2)cc(F)cc(Cl)c1N C1(C(=O)NCC2(O)CN(C(CCN(CCCCC)CC)=O)C2)CCCC12CC2 N1(C(CC2CC(=C)C2)=O)CCC(C(C)CNC(=O)Cc2ncc(C)[nH]2)CC1 C1(NC(C2(N(C)C)CC2)=O)CCN(C(=O)CC(F)(F)F)CC1(C)C C1(CC(=O)NCC(CNC(C2(COC)CC=CC2)=O)CO)CC2CCC1CC2 Cc1cc(C)c(C(N2CCC(NC(=O)CCC3CCCCC3)C(C)C2)=O)c(=O)o1 C=CC(CCC)CC(=O)NCC12CCN(C1)C(=O)C2=O.C1=CC=C1.OC Cc1cnc2cccc(C(=O)NCCOC3CCN(C(C4CCCCC4O)=O)C3)n12 CCCC(CC(=O)N1CCC(NC(N)=O)C1)NC(c1c[nH]c(C)c1)=O c1(C(=O)NCCCN(C(CC(C(CC)C)O)=O)C)cc(=O)c2cc(F)ccc2o1 CCS(=O)CC(=O)N(C(c1ccccc1)C(=O)Nc1ccccc1)C c1(CC)cc(C(N2CCC(NC(c3nnc(O)cc3O)=O)C(C)C2)=O)ccc1Cl C(C(C)(C)CCCO)NC(c1n(C)nnn1)c1nnnn1-c1ccc(OC(F)F)cc1 C(=O)(CCC(N)=O)N1CC(CC(C)NC(C(CC)Oc2ccccc2)=O)C1 N1(C(c2n(C(C)C)ncn2)=O)CCC(C)(CNC(=O)CNC=O)C1 C(CC(=O)NC(C)Cc1ncc[nH]1)(C(C)C)NC(CCCOC(C)C)=O CCC(C(=O)NCC(=O)NCCC(=O)OCC)C(F)(F)F N1(C(C(COC)N(C)C)=O)CCC(F)(CNC(c2sc(C)cc2OC)=O)C1 c1(C(N2CCC(C)C(NC(=O)CCCn3cccn3)C2)C)ccc(F)c(F)c1 C(CCC(C)C)(C(=O)N(C)CCOCCNC(c1sccc1OC)=O)OC.C1(C)CC1 N1(C(C(CC=C)CC(F)F)=O)CCCC2(CCCN2C(C2CCN(C)C2=O)=O)C1 N1(C(CCCOC(C)=O)=O)CCCC2(CC(NC(c3cnn(C)c3Cl)=O)CO2)C1 c1(C(=O)NCCCN(C(CC=C(C)C)=O)C)cc(Br)c(C)cc1F N1(C(COCCSC)=O)CCS(=O)(=O)C(CCNC(=O)C(=Cc2cccs2)C)C1 N1(C(C(=O)OC(C)C)=O)CCN(C)C(CN(C)Cc2ccc(COC)cc2)C1 C(C(CNC(=O)CCCn1ccnc1)C(F)(F)F)NC(C(c1cnn(C)c1)C)=O C(=O)(CC(C)(C(F)F)N(C)C)N(CCNC(c1nc(C)[nH]c1C(F)(F)F)=O)CC c1(NCc2ccc(N3CCN(C)CC3)nc2)ccc2nonc2c1 N1(C(CC2C(NC(C(C)N3CCCC3)=O)CCC2)=O)CCCCC1C(=O)OC c1(OC)noc(C)c1NC(C)=O.N12CCN(CC1)C(=O)C(C)OCC2=O c1(C(N(C(C)CNC(=O)CCc2cnc(C)o2)CC)=O)ccc(C(F)(F)F)o1 C1(C(N(c2ccn(C)n2)CC)=O)CN(C(C2C3CCCC23)=O)CC12CCC2 c1(C(=O)NC23CCN(C(CC=C)=O)C2CCC3)cc2c(C)cc(Cl)cc2[nH]1 c1(-c2ccc(C#N)cc2)cc(Br)ccc1S(=O)NNc1ccc(Cl)cn1 c1(C(=O)NC(CCN(C(CCC2CC(C)C2)=O)C)(C)C)cc(C#N)c[nH]1 C(=O)(C(CO)C(C)(C)C)NC(CCCNC(c1c(Cl)cn(C)n1)=O)c1cccs1 N1(C(c2n(C(C)C)ncc2Cl)=O)CCN(C(C2CCCCC2)=O)C(C(C)(C)C)C1 C1(C(C2(C3CN(C(C4=NOC(C)C4)=O)C3)CC2)=O)CC12CCOC(C)C2 CCC(C)(C)C(=O)C(=O)N1CC(C(O)C(=O)NCC(c2ccccc2)F)C1 CC1CC(NC(=O)CCc2cnn(C)c2)CN1C(=O)C=CCN(C)C c1(C(=O)NCC2C=CC(NC(c3[nH]cc(C)c3)=O)C2)n[nH]c2c1CC(C)CC2 C(=O)(C(C)(C)CC(=O)OC)NC(C(N1CCC(C=C)CC1)=O)CN(C)C c1(C(=O)Nc2c(C)cc(NC(c3cc(Cl)cn3C)=O)cc2)ccc(S(C)(=O)=O)[nH]1 c1(C(N2CCC(N(C(C3N(S(CCC)(=O)=O)CCC3)=O)C)C2)=O)cnn(C)c1F C(=O)(CC(C)(C)CCC)N(CCCNC(C(CCC)CC1CCCCC1)=O)CC N1(C(C=C(C)C2CC2)=O)CCC2CCN(C(c3ccc(C4CC4)cn3)=O)CC12 C(=O)(C(O)C(C(C)C)OC)N1CC(CC=C)(C(=O)NCCC2CCCCCC2)C1 Cc1nc(Cl)ccc1C(=O)NCC1CCCN(c2cc(O)nc(O)n2)C1 C(c1cccs1)=C(C)C(=O)NCCC(C)NC(=O)CCc1cscn1 CC(CF)C(=O)NC1CCC(CCNC(c2cnnn2C)=O)C1 N(C(=NCC1CCCC1)NCC(n1ccnc1C)(C)C)Cc1n(CCC)nnn1 N1(C(=O)CCc2ccc(Cl)cc2)CCCC2(C1)CN(C(=O)CCF)C2 C1(CC(=O)N(C)CC2CC2(C)C)CC2(C1)CN(C(C1(C)CC3(CCC3)C1)=O)C2 C(=O)(CCCC1CCC1)N1CC(C(C(=O)NC(C2(O)CCOC2)C)C)C1 N1(C(C2(S(C)(=O)=O)CCC2)=O)CC2(CCC(CNC(=O)C=C3CCSCC3)O2)C1 c1(NC(CCOC2CCN(C(c3cnc(CC)o3)=O)C2)=O)cc(C)nc(O)c1 C1(C(=O)NC(c2nncs2)C)CCN(C(c2n[nH]c(O)n2)=O)C1 C1(NC(C(C)=C(CC)C)=O)CCN(C(=O)CCN2CCCC(N(C)C)C2)C12CC2 c1(C(N(CCOCCN(C)CCO)C)=O)cc[nH]c1C.C(C(=O)N)NCCOC c1(C(=O)NC(C(C)NC(c2cccc(CC=C)c2)=O)C)ccc(OC)cc1C c1(COC)nc(C)cc(=NCC(C2CCCC2)NC(=O)CCc2ccccn2)[nH]1 C1(N(C)C(c2c[nH]cc(Br)c2=N)=O)CC2CCC(C1)N2C(c1ccc(F)o1)=O N1(C(C(C)SCC)=O)CCC(F)C(NC(=O)C=C(C)c2ccccc2)C1 c1(CC(=O)NCCC(C)(C)NC(Cc2nc(C)oc2)=O)ccc(OC(C)C)cn1 C1(NC(c2ncccc2Cl)=O)CN(Cc2cc(Cl)cnc2F)CCC1C(F)(F)F c1(-n2ccc(C(=O)NC3CCC(NC(CC4C(C)(C)C4)=O)C3)n2)cccc(C#N)c1 c1(OC)ccc(C(=O)NCC2CN(C(c3ccccc3SC(F)F)=O)C2)c(Cl)n1 C1(CC)CCCN(C(c2cc(O)ncn2)=O)C1C(=O)NCC(C)CC(C)C S(=O)(=O)(c1cc(Br)ccc1Cl)C(c1ccc(NC(CN2CCOCC2)CO)nc1)=O N1(C(CC2CC(NC(c3ccc(C(C)C)o3)=O)C2)=O)CCOC2(CCCC2)C1 N1(C(C2(CO)CCC2)=O)CCC2(CCC(CNC(C3CC(F)(CO)C3)=O)O2)CC1 C1(CCNC(CCn2c(C)ncc2)=O)CCCN(C(=O)C(C)(O)C2CC2)C1 C(=O)(CS(=O)C(F)(F)F)NCC1(NC(CCc2n(C)cnc2)=O)CCCCC1 C(CN=c1cc(C)c(S(=O)(=O)N2CCCC3OCCC23)c[nH]1)Oc1cccc(C)c1 c1(C(N2C(C)CC(CNC(c3c(C)ccnc3Cl)=O)C2)=O)cnc2[nH]cnc2c1 c1(C(N2CC3C(CNC(=O)COc4ccncc4)C3C2)=O)ccc2cc[nH]c2c1 Cc1cc(C(N2CCOCC2CNC(c2conc2C)=O)=O)n(C)n1 c1(C(=O)NCCC(CNC(c2c(CC)cns2)=O)O)cc(N)c(Cl)c(O)c1 N1(C(CSCC#C)=O)CCC(CF)(NC(C2C(c3ccccc3)C2(F)F)=O)C1 c1(CC(=O)NC(CNC(C2C(C)C2)=O)C2CCC2)ccc(N2CCCCC2)cc1 N1(C(c2ccc(OCOC)cc2)=O)C2CCC1CN(C(c1cccnn1)=O)CC2 C1(CNC(CCC(C)C)=O)CC2CCC1N(C(c1cccc(C3(C)CC3)c1)=O)C2 c1(C(=O)NC(CCOC)CNC(C2(COC)CC2)=O)cc2cccc(C)c2o1 Cc1noc(C(F)(F)F)c1C(=O)NCC1(CNC(C2CC2F)=O)CCCC1 CC1CN(C(C2(O)CCCCCC2)=O)CC(C)N(C(=O)CN(C)C2CC2)C1 C1(C(=O)NC(CN(CC(=O)NCCOC)C)C)CC1(F)F C1(NC(CCC)=O)CCC(CNC(=O)CCCc2ccc(C)s2)C1 Nc1ccc(C(N2CCCCC(NC(=O)COCCF)C2)=O)c2ccncc12 C#CCC(C)(C)C(=O)N1CC=CC(C(N2CC=CC(O)C2)=O)C1 N1(C(c2nc(C(C)C)oc2)=O)CCN2C(=O)C(NC(C3(O)COC3)=O)CC2C1 c1(C(N2CC(c3ccc(OC)c(F)c3)(O)C2)=O)cc2ccc(Cl)cc2nc1C c1(C(=O)NC(CC(C)NC(CN(C2CC2)CC)=O)C)ncccc1N(C)C C(=O)(C(C)C(C)(F)F)NCC(CC)(CC)NC(c1ccc([N+](=O)[O-])s1)=O C(=O)(CC(O)CC(C)(C)C)NC(C(=O)NC1CN(CC)C(=O)C1)(C)CO C1(CNC(CCCC(=C)C)=O)CC2CCC(C1)N2C(=O)C(C)(C)S(C)(=O)=O C1(NC(CC2CC(OC)C2(C)C)=O)CC2(C1)CC(NC(C1CN(C)C1)=O)C2 c1(OCC2(CNC(C)=O)CC23CCC3)cccc(C(=O)NOC(C)C)c1 c1(CNC(C(c2cn(C)nc2)=O)=O)ccc(CF)cc1.C1(C=O)(C2CC2)CCCO1 N1(C(CC(CCC)NC(=O)C(C)c2ccsc2)=O)CCn2ccnc2C1 Cc1n[nH]c(C)c1C(=O)NCCC1CSCCN1C(=O)CCCOC(C)C Cc1nc(C)n(CCC(=O)NCCc2cn(-c3ccc(C(=O)O)nc3)nn2)n1 N1(C(c2c(CNC(C(C)CN(C)C)=O)c[nH]n2)=O)CCCCCC1C.NC C1(C(=O)NN(C)C)(N(C)C)CCCC1.c12cc(on1)CC1C(C1)C(C)NC2=O Cc1nc(N(CC(O)CN(C)C(C2(C)CC3CCC2C3)=O)C)c2ccsc2n1 N1(C(c2nc(OC)c(F)cn2)=O)CCC(C2(NC(=O)C=CBr)CC2)C1 Cn1cc(C(F)=CC(=O)NC2CC3CC(NC(=O)C4=CCOC4)C3C2)cn1 N1(C(=O)CC2(CO)CC2)CCN(C(C2CCCCO2)=O)C2CS(=O)(=O)CC12 CC(C)(F)C(C)(F)C(=O)N1CC2C(C(=O)NCc3ccccc3C#N)C2C1 C1(NC(C2CCOC2)=O)CCN(C(=O)Cc2cncnc2)C1c1ccccc1 c1(C(=O)NCC2(CNC(c3cc(O)ncc3Br)=O)CCCC2)cc(Cl)cc(Cl)c1Cl c1(OC)ccc(CCCC(=O)N(C)CCN(C)C(C2SC3C=CC2C3)=O)cc1 C1(n2cc(-c3n[nH]cc3C)nn2)(C(=O)NCC(=C)F)CCNC1=O O=C1CCOC(C(N2CCC(N3CCN(C(=O)CCn4cccn4)CC3)C2)=O)C1 c1(NCCC(C)C)cc(=NCC(Cc2ccc(Cl)cc2)CO)[nH]c(C(F)(F)F)n1 C#CC1(C(=O)NCC(C)(O)CC=C)CN(C(=O)CC2CC(C3CC3)C2)C1 C1(C(=O)NCc2scc(C(=O)NC(C(=O)OCC)C3CC3)c2)CCCN(C)C1 Cc1c(CC(N2CC(F)CC2CN(C(=O)CCc2ccnn2C)C)=O)cnn1C CCC(C)N=c1[nH]c(=NC(C)c2c(Cl)ccc(F)c2Cl)c2ccc(C)cc2[nH]1 c1(C(=O)NC2CC2CNC(c2cnc(Cl)[nH]2)=O)ccc2nccnc2c1 Cc1cc(F)cnc1C(=O)NC1CC1CNC(c1cccc(C2CC2)c1F)=O c1(C(N2CC(CCC)C(NC(=O)C=Cc3ccoc3)C2)=O)cccc(O)c1C c1(C(=O)NC2CC3CN(C(c4sc(F)cc4Cl)=O)CC23)ccc2c(O)n[nH]c2c1 C=CCCC(C=O)Nc1cc(COC)nn1C.C(C(F)(F)F)NC(=O)OC(C)(C)C CCCC(CC)C(=O)N1CC(F)CC1CC(=O)NCc1ncn(C)n1 N1(C(c2c(C(C)C)n[nH]c2)=O)CC2CCC(C1)N2C(C1CC(=O)CCO1)=O CC(C)(O)C#CC(=O)NC(CC1CCCC1)C(=O)NC1CCCCC1 Cc1ncc2cc(C(N3CCC(C)CC3CNC(=O)CCCN(C)C)=O)ccn12 C1(C)(CNC(c2n(CC)cnn2)=O)CCN(C(c2cncc(F)c2)=O)C1 n1(CCC)ccc(=NC(=O)C2CCN(C(c3cnn[nH]3)=O)CCO2)[nH]1 C(=O)(CCC(C)(C)F)NC.CCCCC(CNC(c1cc(C)c(C(=O)OCC)o1)=O)NC C1(CC)(CNC(=O)C(O)C2CN(C(=O)CCNC(C)=O)C2)CCC(=O)N1 C=CCC(CC)C(=O)N1CC(C(=O)Nc2ccc(F)c(CO)c2)CCC1C CCCC(CNC(C1(C)CCNC1=O)=O)C(=O)NC(c1cnccc1C)C C1(CNC(c2c(C)ccnn2)=O)CC12CCN(C(=O)C=Cc1ncc[nH]1)CC2 N1(C(c2cc(SC)oc2)=O)CCOC(C(N2CCCC2(C(C)C)CO)=O)C1 c1(C(C)NC(=O)CCNC(C2C3COCC23)=O)ccccc1F N1(C(c2c(CNC(C3CCCCC3)=O)cc[nH]2)=O)CC2(CC2)CC1CN1CCCC1 CCCCCCCCC(F)C(=O)NC12COC(NC(=O)C(C)S(N)(=O)=O)(C1)C2 C(=O)(C(C)CC(F)F)NCC1CCN(C(c2c(C)onc2-c2ccncc2)=O)C1 C(=O)(C(C(C)(C)C)NC(C1CC(OC)C1)=O)Nc1ccc(OCC)nc1 c1(CC)oc(C)cc1C(=O)NC(C)(CO)C(=O)N1CCC(C(C)(C)O)C1 c1(C(=O)NC2CC3CN(C(CSC(C)(C)C)=O)C2C3)cnc2[nH]cnc2c1 CC1(NC(c2cnc[nH]2)=O)CCN(C(C2CCCN2N=O)=O)CC1 N1(C(C(C)C2CC2)=O)CCC(O)(C(C)NC(=O)Cn2cc(CN(C)C)nn2)C1 CC(C)C(C(=O)OC(C)(C)C)C(=O)N1CCC1NC(c1ccc(C(N)=O)cn1)=O C1(C(=O)NC(C2OCCN(C(C(CC=C)(C)C)=O)C2)C)CCCC2(CCC2)C1 c1(CC(N2CC(C)(NC(Cc3ccc(OC)cc3)=O)C2)=O)ncn2c1CCCC2 c1(C(N2CC(CNC(C3(CSC)CC3)=O)C(C)C2)=O)c(C)cc(C)cc1N N1(C(C(C=C)O)=O)CCCC2(CCN(C(c3cc4c[nH]nc4s3)=O)CC2)C1 CC1C2=C(C(=O)N1C)C(c1cccc(C(N)=O)c1Br)NC(=O)N2CC1C(CO)C1 c1(CC)nccnc1C(N1CCC(O)(CNC(=O)CC2CC(OC)C2)C1)=O C1(O)(CCNC(CCOCCC)=O)CN(C(=O)CC(c2ccccc2)N(C)C)C1 c1(OC(C)C(N2CCNC(c3ccncc3)C2)=O)cccc(F)c1F O=C(C1=CCN(C(C2CC=CC2)=O)CC1)NC1CCOC1 N1(C(C(C)CF)=O)CC2CC1CN(C(=O)CSCc1nc3ccccc3[nH]1)C2 c1(C(=O)OC)ccccc1C(N1CC2CC2(CNC(c2cc(C)no2)=O)C1)=O c1(C(N2C(CNC(CCC)=O)CC(C)(C)C2)=O)cc2cc(Cl)ccn2n1 c1(C(C)C)ccc(C(N2CC(F)CC2CNC(=O)CS(=O)(=O)N(C)C)=O)nc1 C(=O)(CC(C)(C)C(=O)N1CC2(CCC2NC(C2CCC(=O)N(C)C2)=O)C1)OC N1(C(=O)NC(c2ncccn2)C)CCCN(C23CCCC2C3)CC1 N1(C(c2c(C)nns2)=O)CCN(C(c2ccc(I)c(Br)c2)=O)CC1CO C(=O)(C#CC(C)(C)C)NC1C(OC)CN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C1 CCS(=O)(=O)CC(=O)NC1CCCCN(C(c2cncc(NS(C)(=O)=O)c2)=O)C1 N1(C(C2(c3ccc(C)o3)CC2)=O)CC2CC2C1.C(=O)(O)C(=O)O c1(CC(=O)N(CCC)CCNC(=O)C(=O)N(C)C)ccc(N(C)C)cc1C C1(C(N2C(CCC)COCC2)=O)COCCN(CCOC2CC2)C1 N1(CC(=O)NC(=O)NC(COC)C)CCCC(Cc2oc(CO)cc2C)C1 N1(C(CCN(CCC)C)=O)CCN(C(=O)CC(C)C(C)(C)C)C2CCC12 C1(NC(C(C)SCCCC)=O)CCN(C(=O)C(c2cn(C)nc2C)O)CC1O c1(C(NOCCC=C)=O)ccc(CNC(C2(C#N)CCOC2)=O)cn1 CC1(C)C(NC(c2nocc2C2CC2)=O)CCN1C(=O)CC1CCCCC12CC2 C(=O)(C1=CC2CCCC12)NC1CCC(F)(CNC(c2c(COC)scc2)=O)C1 c1(CC)ccc2c(C(C)(C)C(=O)CNC(=O)OC(C)(C)C)cc(=O)oc2c1 c1(CC(C(=O)NC(CN(C(CC2(C=C)CCC2)=O)C)CC)O)c(F)cccc1F N1(C(C(CC=C)NC(C)=O)=O)CCC2(CC2)CC1C(N1CC2(CCCC2)C1)=O Cc1cc(O)c(C(=O)NC(C)(CNC(c2ccc(Cl)nn2)=O)C2CC2)nn1 C(=O)(CCS(=O)(=O)Cc1cccc(C)c1)N1C2C(CNC(C(CC#C)C)=O)C(C2)C1 C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CCN(C(=O)C=Cc2nccs2)CCC1CO c1(C(N(C2CC(NC(CC3CC(C)C3)=O)C2)C)=O)ccc(S(=O)(=O)CCO)cc1 N1(NC(NCC(=O)NC)=NCC2CC(=CC=C3CCC3)C2)CCC2C(C1)C2(F)F CC(CC(=O)NC(C)CCNC(c1ccc(C#N)s1)=O)CC(C)(C)C C(=O)(C1CCCc2c1ncn2C)N(C(C)CNc1cc(C(F)F)ncn1)C C1(C(=O)NCC2(C(F)F)CCN(C(C3(Cl)CC3(F)F)=O)C2)(OC)CCCOC1 C(CNC(=O)CC1(CO)CC1)(C(C)(C)C)NC(Cc1cn(CC)nn1)=O CCC(CC)C(C)C(=O)N(C(CC)CC(=O)NCC1CC(C)=NO1)C N1(C(C2CN(C(C3CCCS3)=O)CCO2)=O)CC2COCC2C1 C1(C(=O)N)CCCCC1C.c1(C(C)CC(=O)CSC(F)(F)F)nncn1C C1(C2CCCN(C(=O)Cc3ccco3)C2)(NC(=O)Cn2cc(F)ccc2=O)CC1 N12CCOC(C1)C2=O.C12(NC(C3(CC=C)CCC3)=O)CC(COC)(C1)C2.C=O C1(C(N(CC(C)C(=O)NC(C)C2CC2)C)=O)C2CCC(F)C12 C1(C(C)C)CCCN(C(=NC(C)CN(C)C)NC2CCOCC2)C1 C1(Cn2cc(C(C)(C)SC3CCN(O)C3=O)nn2)CCN(C(N)=O)CC1(F)F C1(CN(C(C2CC2F)=O)CC)CCCCN1C(=O)C=Cc1ccc(C2CC2)o1 c1(NC(c2n[nH]c(C)c2C)c2n(C(C(=O)OC)C)nnn2)cn(C)nc1C N1(C(c2cc(C)ncc2)=O)CCC(CNC(C2OC(C)CC2C)=O)CC1C C1(NC(c2c(CC)onc2)=O)(CO)CCN(C(C2CCC(C)(C)CO2)=O)CC1 C1(NC(C(CC)NC(C=CC(CC)C)=O)=O)CCCC(CC(=O)NC)C1 N1(C(COCC=C)=O)CCCC(CO)(CNC(C2CCC(=O)N(C)C2)=O)C1 c1(C(N2CCC(c3cccc(OC)c3)C2)=O)nn(C)c2c1CS(=O)(=O)CC2 C1(O)(C(N2CC(CC=C)(NC(=O)CCC3C(=O)NN=C3C)C2)=O)CCCCC1 c1(-c2cn(C3CN(C(=O)C(O)c4ccsc4)CC3O)nn2)ccn2ccnc2c1 N1(C(CSc2n(C)nnn2)=O)CCC(O)(CCNC(c2csc(O)n2)=O)CC1 C1(O)(CC(=O)NC(C)(C)CC2CCCC2)CCN(C(C2CCC(F)CC2)=O)CC1 c1(C(N(CC(CNC(Cc2c(C)n[nH]c2C)=O)C)C)=O)ncn2cc(Cl)ccc12 C1(NC(C(C)NC(=O)C2CC2)=O)CCN(C(c2cncc(O)c2Cl)=O)CC1CO c1(CC(=O)NCC2CN(C(C3CCC(C)(CC)O3)=O)C(C)C2)cc(C)cc(F)c1 O=C(CC(C(F)F)NC(C1(O)CCOC1)=O)Nc1ccc[n+]([O-])c1 Cc1ccc(F)c(C(=O)OCCN2C3CC2CN(c2nccc(OCF)n2)C3)c1 CC(C)CC(O)C(=O)Nc1c[nH]nc1C(=O)Nc1ccc(-n2cccn2)nc1 C1(CCCC)CN(C(c2cc(OC)ns2)=O)CCN1C(c1cnc(OC)s1)=O N1(C(N(C(C(CC)C)C)C2CC2)=O)CCC(C2CC2(F)F)C1 c1(NC(CCC2N(C(C(CCC)N(C)C)=O)CCCC2)=O)cccn(CC)c1=O N1(C(C2(SCC)CC2)=O)CCC(CF)(NC(=O)C(C)C2CCCC2)C1 C1(C(=O)OCC)CN(C(=O)Nc2ccc(F)c(-c3ncco3)c2)CC1C1CC1 C1(CNC(C(COC)(C)NC(=O)CCCc2cccs2)=O)CCn2cncc2C1 c1(C(=O)NCC2(OCC)CN(C(=O)C(C)=C(C)C)C2)cc2ccc(CC)cc2[nH]1 Cn1nc(C(=O)NC2C3CC2N(C(c2c[nH]c(N)c2)=O)C3)c2c1CCC2 C1(COC)(NC(=O)C(c2cscn2)N(C)C)CCN(C(=O)CN(C)C)CC1 C1(C(N2C(C(=O)NCCC(C)O)(COC)C=CC2)=O)OCCCC1(C)C S(=O)(=O)(CC(=O)N1CC(c2cn(-c3nccnc3N)nn2)(NC(C)=O)C1)NCC C(C(C(F)(F)F)N1CCN(C(=O)C(C(C)O)N(C)C)CC1)NC(CC=CCC)=O C(=O)(C(F)C(C)(C)O)N(CCCNC(C1CC(=C(F)F)C1)=O)CC N1(C(COCCC(C)C)=O)CCC(O)(NC(=O)C(C)OCCN(C)C)C1 O=C(CCCc1nccs1)NC1CCC1CNC(=O)CC1CCC(C2CC2)O1 Cc1ccc(C(C)C(N2CCC(O)(CCNC(=O)C=Cc3cc[nH]n3)C2)=O)cc1 C(c1cc(F)cc(F)c1)=CC(N1CC(OC)C(NC(=O)C=CC2CC2)C1)=O N1(C(C(C)OCC=C)=O)C2CCC1CC(CNC(=O)CCc1ccnc(C)n1)C2 C1(=O)C2=CC(O)C(C2)N1.n1(CC)ccnc1CN(C(=O)CN(C1CCC1)C)C c1(C(N(C(c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)C)C)=O)cn(C)ccc1=O c1(OC)ccc2c(CC(N3CCN(c4cnccn4)C(C#N)C3)=O)coc2c1C C(=O)(CC(=O)NCCCCC1CN(C(C23CSCC2C3)=O)C1)NCC C#Cc1cnn(C)c1C(=O)NC1CC(NC(c2cnc(OC)s2)=O)CC1O c1(C(=O)NCC(C)CO)nnnn1CC(F)(F)F.C12(CC1)C(=O)N2.NC(=O)NC Cc1cc(C(N2CCCC2Cn2cc(COC3CCCCO3)nn2)=O)cc(C)n1 c1(NCCCC(=O)NCC(CC)NC(C2CCOCC2)=O)cncc(C)n1 N1(C(CCC(C)(F)F)=O)CC(NC(=O)COc2ccc(O)cc2)CC12CCC2 C(=O)(CC(Cc1ccccc1)CC)NCC1(F)CN(C(CC(CC)C)=O)C1 c12nccc(n1)NC2c1nnnn1CCSC.C(=O)(CCCOCC)OCC C1(C(=O)NC(CC#C)C(=O)OC)CC2(C1)CN(C(c1ccnc(Cl)c1C)=O)C2 Cc1cc2n(n1)CCN(C(C1CC(NCc3c(Cl)cc(F)cc3Br)C1)=O)C2 C1(NC(C2N(CC)CC2)=O)CCN(C(c2noc(C(C)C)c2C)=O)CC1O CC1(C(=O)NC2CC(CC(N3CCC3C(N)=O)=O)C2)CCCO1 c1(C(c2nnnn2CCC2CC2)NC2(CC=C)COC2)ccc(N(C)C)nc1 N1(C(C2(C)CC(=C)C2)=O)CC2(CCCN(C(C3CC(C4CCCC4)C3)=O)C2)C1 C#Cc1ccc(F)c(C(=O)N(CCC(C)NC(c2c[nH]cc(C)c2=O)=O)C)c1 N1(C(c2occ(C)c2)=O)CCCCC1C(C)NC(c1cc(Br)cn1C)=O N1(CC)C(=O)C=CC(C)N(C)C(=O)C(C)(OCC)C1CC Cc1cnccc1-c1cn(C(C)C(=O)NCC2C3CCC23c2ccccc2)nn1 C1(C(=O)NCC2(C)N(C(C(n3ncc(C)c3)C)=O)CCC2)CCOC(=O)CC1 Cc1ccc(SCC(N2CCC(OCCNC(C3C4CC5C(C4)C35)=O)C2)=O)cc1 CC(C)(O)C#CC(=O)N1CCN(CC(=O)NCc2cc(C3CC3)ccn2)CC1 O=C(C1CCCc2nn[nH]c21)NCC1CN(C(=O)C=C(Cl)Cl)CCO1 c1(CNC(C(n2cc(-c3cn(CCOC)nc3)nn2)C)=O)cc(Cl)c(Cl)n1C CC1(F)CCCN(C(=O)CCN(C(c2cncc(O)c2)=O)CC2CC2)C1 N1(C(CCC(=O)NCC)=O)CC2CC1CN2C(=O)Cc1cccc(OC)c1F C(CC(C)(C)CC(=O)N(CCNC(=O)CN1CCOCC1=O)C1CC1)OC c1(OC2CN(C(C(=O)OCC)=O)C2)ccc(CNC(C2CCCOC2C)=O)cc1 N1(C(=O)OC)CCN(C)C(c2ncc[nH]2)C1.C1CCN1S(C)(=O)=O CC(C)(C)CCC(=O)N1CCCCC1N(c1nnc(C2CCCO2)s1)C CC1CN(C(=O)CC2CCC(=O)N2C)CC1CNC(=O)C(C)Cn1ccnc1 C1(CC)(COC(N2CCN(C(=O)OC(C)(C)C)C(C)C2)=O)CCC(F)(F)CC1 C=C(CN1CCOCC1c1ncon1)C1CCOCC1 C#CCCCC(=O)NC1CCC(CNC(c2cc(C)c(CC)s2)=O)C1 C1(NC(c2cc(CC)sn2)=O)(CSC)CCCN(C(=O)C(C(C)C)N(C)C)C1 c1(C2CC(C(=O)Nc3cnc(C)n3C)C2)ccc(N2CCN(C)CC2)c(F)c1 N1(C(C23C(NC(c4n(C=C)ncc4)=O)CC(CC2)C3)=O)CCC(C#N)CC12CC2 C(CNC(=O)C(c1ccnn1C)C)(CC(F)(F)F)NC(CCCNC(=O)OC)=O N1(C(c2c(OCC)cccc2)=O)CCC2(CCN(C(=O)C(COC)OC)CC2)C1 C(=O)(C1=CCN(C)C1)NCCC1CCCN(C(C(CCC)OCC)=O)C1 N1(C(CC2(COC)CC2)=O)CC(NC(=O)CCS(N)(=O)=O)Cc2ccccc21 C(=O)(C1CCc2c[nH]nc21)NC1C2CN(c3nc(OCC)c(Cl)cn3)CC21 C1(n2cc(CNC(=O)OC(C)(C)C)nn2)(CN(C)C)CCOCC1 c1(OC(C(=O)NCC2N(C(C(F)=CC)=O)CC=C2)C)ccccc1Br CC1CN(C(c2cnc(S)n2C)=O)CCC1CNC(C1CC(C)(O)C1)=O N1(CC#N)CCCC2C1CCN2C(c1cocn1)=O N1(C(COCCCOC)=O)CCCC(C)C1CNC(c1nc(Cl)sc1C)=O C=CC1(C(=O)NC2CC(O)C23CCC3)CCN(C(=O)CCC(C)(F)F)CC1 c1(OC)cccc(C(N2CCC(CNC(C3CCC(C)CC3)=O)C2)=O)c1 C(=O)(C(CC(C)C)CC(C)C)NCCC1N(C(CC(CC)C2CC2)=O)CCCC1 C12(OC)CCC(NC(c3ccn(CCNC(c4cnc(O)o4)=O)c3)=O)(CC1)C2 n1(CC)c(C)cc(C(N2CCC(NC(c3nn[nH]c3Cl)=O)C2C)=O)c1C C1(C(=O)NC2CC(C)(NC(C(CC)OC3CCCC3)=O)C2)CC1C1CCC1 CS(C)(=O)=NCC(=O)N(C1CCN(C(=O)Cn2cc(C#N)cn2)C1)CCO C(C1=CCN(C(C2CNC(=O)N2C)=O)CC1)NC(c1cn(C(C)C)nn1)=O Cc1onc(C(=O)NC2CCCCC2N(C)C(c2cnc(O)s2)=O)c1[N+](=O)[O-] C12(NC(c3ccc(OC)cc3)=O)CCCC1N(C(=O)C=C(C)C(F)F)CCC2 C1(C(=O)NC2C(NC(c3cn(C)nn3)=O)CCC2)CC(C)(C)CC(C)(C)C1 C1(C(=O)NC2CCC(C(c3nn[nH]n3)N)C2)CCCN2CCCCC12 CN(CCc1nc2ccccc2s1)N1CCCC(O)(CO)C1 C1(NC(=O)C=C2CC2)CC2CN(C(c3cc(-c4ccncc4)ccn3)=O)CC2C1 N1(C(c2ccc(C)s2)=O)CC2CCC2(NC(=O)C(C(C)C)NC=O)C1 c1(OC)ccccc1C(=O)NCC1CC2CC2N1C(c1ccoc1)=O C1(OCC)CC2(C1)CC2C(N1CCSCC1CCNC(C1(C)CCOCC1)=O)=O C1(C#CC(=O)NCC2CCOC2C(=O)NCC2CCOC(C)(C)C2)(CC)COC1 C1(NC(CCC)=O)CCN(C(c2cccc3c2C2CCC3O2)=O)C12CCCC2 C1(NC(C2N(C(C3N(C)C(=O)OC3)=O)C(C)CC2)=O)CCC12CCCC2 C(=O)(C1SCCc2sccc21)NCC1CN(Cc2cn(C3CCN(C)C3)nn2)C1 Cc1[nH]nc(C(=O)NC2CC(CNC(=O)C(c3ccc(F)cc3)(C)F)C2)c1C C1(C(=O)NCC(CC)NC(=O)Cc2cc(C)[nH]n2)C2CCC3C(C2)CC13 c1(NC(CCC=C)C)[nH]c(=NCCCCF)nc2c1cnn2C(C)C CC(CS(C)=O)C(=O)NC1CC(C)(NC(=O)COCCCc2nccn2C)C1 CC1(c2cn(C3CC3)nn2)CCCCCC1.C12CCC(CC1)NC(=O)C1CC(C1)N2 C1(n2cc(CCN(C)CCOC(F)F)nn2)CCCN(C(N)=O)C1.CO CCC(C)(C)C(O)C(=O)N1CC(CNC(C2CC3CCC(C2)S3)=O)(COC)C1 C1(NC(C2(CC)CC2)=O)CN(C(=O)C(C)(C)Cc2ccc(Cl)cc2)CCC1CO Cc1cccc(C(=O)NC(CNC(C2(O)CC2)=O)C(C)C(C)C)c1C CCC(CC)(CC)C(=O)N1CCC(NC(c2coc(C3CCC3)n2)=O)C(C)C1 c1(C(N(C2CCN(C(CC(COC)C)=O)C2)C)=O)coc(S(=O)(=O)N(C)C)c1 c1(CNc2c(C(N3C4CCC3CC(O)C4)=O)scc2)cnc2ccccc2n1 N1(C(C(c2ccc(OC)c(Br)c2)=O)=O)CC2CC3CC2C1C3O c1(C(=O)NCC2N(C(Cn3ncc(C)c3)=O)C3C(C2)C3)ccc(C(C)C)c(Cl)c1 C1(NC(CCN(C)CC)=O)CCCOC12CCCN(C(c1cc(C)n(C)c1)=O)C2 Cc1cc2occ(CC(=O)NC3CC(CNC(=O)COCCF)C3)c2cc1C N(C(=NCc1cn(CC2CCOCC2)nn1)NCC(C)(C)C)C(COC)C c1(C(=O)NCC(CC)Nc2ncc(C(F)F)cn2)cc([N+](=O)[O-])ccc1Cl C12(C(N(C(CC)C3CC3)C)=O)CCCC1N(C(=O)C(C(C)CC)NC(C)=O)CCN2 N1(C(C2C(C)(C)COC2)=O)CC2(CC2)CC1CNC(C1CC=CCC1)=O C12CC3CCC(C1)N3C(=O)C(OC)NC(=O)CC(C)CN2C1CC1.CC.OC c1(C(N(C(C(=O)N(CC(C2CCC2)OC)C)C)C2CC2)=O)ccnc(C)c1N C1(C)(C(N(C)CC2(C#N)CC2)=O)CCCN1C(=O)CC(F)(F)F CC(CN(C)C)CCC(=O)N1CC2(CCC2CNC(=O)CCCC(N)=O)C1 C1(CC(=O)NCCC(C)N(C(C2C(=C)CC2)=O)C)CCCS(=O)(=O)C1 c12cccc(c1O)C(=O)N2.C1(C(c2ccccc2)C#N)CCS(=O)(=O)C1 c1(C(=O)NCC(CNC(C2(CCCC)CCC2)=O)O)sc2cncn2c1C N1(C(CCC)=O)CC2CC1CN(C(c1cc(Br)c(CC)s1)=O)C2 C(CCCCC(=O)N1CCOC(CF)C1)N(C(=O)CCC(C)N(C)C)C CN1CCCc2c1nn(C)c2NC(=O)NCc1cnc(C(F)(F)F)nc1 C(C(C(=O)NOCC(C)(C)C)NC(c1nc(Cl)cs1)=O)N(C)C CC1(C(N2CCCC(NC(c3cc(O)ncn3)=O)CC2)=O)CCNC(=O)C1 CCCC(C(=O)NC(CCNC(C1C(C)C1C)=O)C(C)C)C(C)C C1(CNC(C2CCCCCC2)=O)CC2(CCC2)CN1C(C1COC2COCC12)=O C1(NC(CC(C)(C)C(C2(C)CC(C)(C)C2)=O)=O)CCCC(C(=O)NC)CC1.CO CCCC(C(=O)NCC(c1ccccc1)CNC(c1cc(Br)no1)=O)OC N1(c2nc(NC3CCN(C4CCOCC4)C3)cc(C)n2)CCC2CCOC2C1 C(N=c1[nH]c(=NC)[nH]c(=NC(C)c2ccc(Cl)c(C)c2Cl)[nH]1)C1(S(CC)(=O)=O)CC1 c1(C(=O)NCC2CCCOC2)cc2n(n1)CCN(C(c1cc(Br)ccc1I)=O)C2 C(=O)(CC(C)CC(=O)N1CCC1CNC(C1CC2CCC1CC2)=O)OC C1(N(CCC)C)CCC2(CCN(C(=O)C(N)CN)CC2)C1 C(CCSC)(C(=O)N1CC(NC(c2conc2C(C)C)=O)CC1C)OC c1(CC)cc(Cl)c2n[nH]cc2c1.C1(C)(CSCC)CCC(NC(C2C3CCN32)=O)CC1 CCC(COC)C(=O)NCC1CC(NC(=O)CC2CCC(=O)O2)C1 c1(C(C)N(C)C(C(Cc2ccco2)CO)=O)noc(C2CC2)n1 c1(C(=O)NC(C2CC2C2CC2)(C)C)cc(Br)c(CN)s1 N1(C(c2nc(CC)sc2)=O)CCC(NC(=O)Cc2cnccc2C)C(CO)CC1 C1(c2nc(-c3cccc(F)c3)nn2-c2cccnc2)CCCc2ccccc21 C1(OC(C)(C)C)CCN(C(c2occc2F)=O)CC12CC2 c1(C(N(CC(O)CN(C)C(C2(N(C)C)CCCC2)=O)C)=O)cc(N)c(F)cn1 N1(C(=O)CSC(F)F)CC2(CC(C(N3CCC3CN=[N+]=[N-])=O)CO2)C1 CCC(C)N(OC)C(=O)c1cccc(CNC(c2ccn(CCF)n2)=O)n1 C(=O)(C(CC)C(C)C)NCCC1CC(NC(C2N(S(CC)(=O)=O)CCCC2)=O)C1 C1(NC(c2c(C(C)C)nn(C)c2)=O)CC(C)CN(C(c2csc(C#N)c2)=O)C1 c1(C(N2C3C(CNC(CC(CCC)O)=O)C(C3)C2)=O)cc(Cl)c(F)cc1F Cc1cc(N(C(=O)CC(C)C(F)F)C(C2CC(C3CC3)=NO2)=O)c(O)cc1F c1(NC(=O)Cc2csc(=NCc3ccc(O)c(F)c3)[nH]2)cc2c[nH]nc2cc1F N1(C(C(CO)OC)=O)CCC2CCCC12C(=O)NC1CC(C(C)O)C1 N1(C(=O)Cc2ccc(CO)cc2)CCOC(C)C1.c1(C2(CO)CC2)cncc(Br)c1 C1(CNC(=O)C=CC2CCOCC2)CCCC(NC(=O)CC2(O)CCOC2)C1 N1(C(CCCC(C)=O)=O)CC2CC(NC(C3CNC(=O)C(C)(C)C3)=O)CC1C2 c1(C(N2C(COC)CN(C(C3CC3C3CC3)=O)CC2)=O)ccn2c1CCCC2 C1(C(=O)NCC2(NC(c3cc(-c4cn(C)nc4)[nH]n3)=O)CCC2)CCC(F)(F)C1 C(=O)(CC(CNC(=O)C(C)(C)C(C)(C)O)CC(C)C)OCC C1(CNC(C2N(C)C(=O)NC2)=O)CN(C(=O)Cn2cc[n+](C)c2)CCCO1 O=C(N=c1cc2n([nH]1)CCNC2=O)Nc1ccc(CNS(=O)(=O)C(F)F)cc1 N1(C(C2CC=CC(NC(CCc3cc(C)on3)=O)C2)=O)CC2(CCCC2)CC1C c1(C(N2C(C(C)NC(c3cn(CCCC)nn3)=O)CCC2)=O)cc(=N)[nH]c(Cl)n1 C1(N(C(=O)CSc2n[nH]c(O)n2)C)CCCN(C(c2cc(Cl)ncc2N)=O)CC1 N1(C(=O)NC2CCC(C)(C)OC2)CCn2ccnc2C1 c1(CN(C(=O)C(c2ccoc2)NC(=O)CNC=O)C)cn[nH]c1 N1(C(c2ccc(CC)o2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1CO C1(C(=O)NC2C(NC(=O)C=Cc3ccccn3)CCCC2)CCCCCC1(F)F Cc1ccc(CC(C)CN(C)C)cc1.c12cn(nn1)C1CN(C1)C(C)C(=O)NC2 C1(C(=O)NCc2c(C)ccs2)CCC(C)N1C(c1ccc(C(N)=O)cc1)=O Cc1nc(C(N2CC=CC(NC(C3C(C)C3C)=O)C2)=O)c(C)o1 C1(N(C(=O)C(C)(C)SC)CC)CCCN(C(C2CC(F)(F)C2)=O)CC1 C1(F)(CNC(C2C(CCC)C2)=O)CC(N(C(C2CCC2(C)C)=O)C2CC2)C1 C12(NC(C3(C)C(CC)CCC3)=O)CCC(CO)(C1)OC21CN(C(=O)C(C)(C)C)C1 N1(C(c2cnn(-c3ccccc3)c2)C(=O)NC(C)C)CCC(C)C(CN=[N+]=[N-])C1 c1(CN(CC(N2CCC(C(F)(F)F)C2c2cccnc2)=O)CCO)ccc(F)cc1 N1(C2CN(C(c3ccc(OC(F)F)nc3)=O)C2)CCN(C(=O)C(O)C2CC2)CC1 C1(C(=O)Nc2ccc(OC)c(Br)c2)COC2(C1)CN(C(=O)CN(C)C(C)C)C2 CC1(C(=O)OCCc2ccon2)CC2CCC(C1)S2(=O)=O N1(C(c2cc(=NC)[nH]cc2)=O)CCCC2(NC(C3CCC3OC)=O)CCCC12 c1(OC)cc(C)ccc1CCNC(=O)CN1CCCC(NC(=O)OC(C)(C)C)C1 C1(CC(N2C(C)C(NC(=O)Cc3cccs3)CC2)=O)CCCC2(CCC2)O1 N1(c2ccnc(SC)n2)CC2(CC2)CC1CNC(=O)C(c1ccc(Cl)nc1)(C)C C1(O)(C(=O)NC(CNC(CCN(C(C)=O)C)=O)C)CCOC1 C(C(C)CC(=O)N1CC(CC(C)NC(=O)CC23COC(C)(C2)C3)C1)OC c1(C(N2CCC(C)(NC(c3cc(CO)[nH]n3)=O)C2)=O)ccc(=O)n(C2CC2)c1 N1(C(c2nc(CC)sc2N)=O)CCC(CO)(NC(c2cc(C)nn2C)=O)CC1 Cc1cccc(CC(=O)NCc2cn(-c3ccc(OC(F)(F)F)cc3)nn2)c1Cl Cc1c(C(=O)NCC2(NC(c3ccc(F)s3)=O)CC2)ccc(F)c1F CCC(O)C(=O)N(CCC(c1cccs1)NC(=O)C(C)n1cccn1)C c1(NC(C2C(O)CCN(C(C(CC=C)OC)=O)C2)=O)cnc2n1CCOC2 C(C)(C)(CC(=O)N1CCC(CCC(N2CCCCCC2)=O)C1)OC c1(C(N2C(C3CCN(C(COCCC)=O)CC3)CCC2)=O)cc2n(n1)CCCO2 N1(CCNC(=O)CN2CC3CC3C2)CCC(CSC2CCSC2)CC1 C12(C(=O)NCC(CO)NC(c3cc(N)c(Cl)cc3)=O)CC3CC(C(=O)N1)C2C3 CC(C)CC(CNC=O)CC(=O)NC(CC1CC1(F)F)C(=O)O C12(CNC(=O)C(C3CCCCC3)O)CC(CO1)N(C(c1ccnc(CO)c1)=O)C2 C#CC1CCCN(C(C2(NC(=O)Cc3nc(=N)[nH][nH]3)CCCC2)=O)CC1 c1(OC)cc(-c2cncnc2C(=O)Nc2ccc(C)c(Cl)n2)cc(C)c1 N1(C(CC2(OC)CC2)=O)CCC(CO)(CNC(c2oc(C)nc2C(F)F)=O)C1 C=CCCC(C(=O)N1CCC(CN=[N+]=[N-])CC1)NC(C1CCOC1C(C)C)=O C(C)(CC(=O)N(C)CCN(C)C(c1cnn(C2CCCCC2)c1)=O)SC CC(C)CC(C)(O)C(=O)NC1CCN(C(C2CC3CCC(C2)S3)=O)CC1 c1(OC)ccc2nc(C(c3nnnn3C3(C)CC3)NCC(C)F)sc2c1 C=CC1(CC(=O)NCCCNC(=O)C=CC2(C)CCOCC2)CCOCC1 C1(C(=O)NCC(CC)NC(c2c(Br)noc2C)=O)CC2C=CC1C2 CC(C)C(C)C(CNC(C1(S(N)(=O)=O)CC1)=O)NC(=O)C=Cc1cnn(C)c1 C(=O)(C#CC(C)(C)C)N(C1CN(C(=O)C(C)(C)n2cccn2)C1)C.C1(N)CCC1 C1(C)(C(N(CCCN(C(C(C)OC2CCOC2)=O)C)C)=O)CCN(C)CC1 C(=O)(C=C1SCC(=O)N1C)N1CC2(OCC(NC(C(C)C3CCC3)=O)C2)C1 Cc1cc(C(=O)NC2CCCC2CNC(c2n[nH]cc2Cl)=O)cc(C)c1C C1(CNC(=O)CC(C)C2CCCCC2)CCC(OC)CC1.C(C(C)(C(=O)OC)O)CC C(=O)(C(C)(C)C(N)=O)NC1C(NC(c2c(C(=O)OC)coc2)=O)CCC1 c1(C(=O)NC(C)CC(O)c2ccco2)ccc(-c2cc[nH]c(=N)c2)cc1 c1(CNC2CC(NC(c3c(Cl)cc(C)cc3Cl)=O)C2)cc2ccc(Br)cc2s1 CC(C(=O)N(C)CCc1ncc[nH]1)N(C)C N1(C(Cc2c(C)nn(C)c2C)=O)CC(NC(=O)COCCF)CC(C)(C)C1 c1(C(CNCC(C)CNC(=O)OC(C)(C)C)O)cncc(Br)c1 C1(CNC(COc2c(C)occc2=O)=O)COC(C)(C)CN1C(=O)C1=CCC1 c1(C(=O)OCC)cc(OC)cc(NC(=O)C(O)C(C)SC)c1 c1(C(=O)NC2(CNC(C(C)C(F)(F)F)=O)CC2)nnc2n1CCCCC2 N1(C(CCCC(=O)OC)=O)CCC2CCN(C(c3csc(C(N)=O)n3)=O)CC2C1 C1(OC)CCN(C(C2CCN(C(=O)CCCC#N)CC2)=O)CC1F n1(CCOC)nc(-c2nc(-c3ccc(OC)cc3)nn2C2CCOC(C)C2)cc1C C(C(=O)N1C(C(=O)NCc2cnc[nH]2)CCC12CC2)(C(C)(C)C)N(C)C C1(C(CNC(c2c[nH]c(C(N)=O)c2)=O)NC(C(C)N(C)C)=O)CCCCC1 N1(C(C=CCCC)=O)CC(C)(C)CCC1CNC(=O)CCCS(C)(=O)=O N1(C(C(c2ccc(C)s2)C)=O)CCC2CN(C(=O)CCC3CCCCO3)CC2C1 c1(-c2ccc(CC)cc2)ccc2nc(C(N3CC(C)(O)C(O)C3)=O)cn2c1 Cc1o[nH]c(=NC(=O)C2CCCn3c(C)cnc32)c1C c1(CCC2N(C(=O)CCS(C)(=O)=O)CC(CC)OC2)ccc(N)c(C(=O)OC)c1 N1(C(=O)C=C2CCC2)CCC2C(CCN2C(c2ccc3ncnn3c2)=O)C1 N1(C(CCOC2CN(C(CCCCC(C)C)=O)C2)=O)CCCCC1C1CCC1 C(=O)(CN=c1cc(C)[nH]c(=NCc2cc(N)ccc2F)[nH]1)N(C)CC S(=O)(=O)(c1ccc2c(c1)OCCO2)N1CC(C(N2CC(O)CC2CO)=O)NCC1 CC1(C)C(C)(C(N2CCC(CNC(=O)C(C3CCS(=O)(=O)CC3)O)C2)=O)C1(C)C C1(CCC)CCCN1C(=O)C=CCNC(=O)CC1CCCN1C CCC(C(=O)NC(c1ncn(C)n1)CC)NC(C)=O C(=O)(C(C)(C)CC(F)F)NC1CC(C)N(C(=O)C=Cc2ccc(O)cc2)C1 N1(C(c2cnc(C(F)(F)F)cn2)C(=O)NCC=C)CCOC(C(F)(F)F)C1(C)C C1(C)(C(=O)NCC23CC(NC(C4C(C(=O)OC)C4)=O)(C2)C3)CCN(C)C1=O N1(C(c2ccc(Cl)cc2-c2ccccc2)=O)CCCC(C2CCNCC2)C1 c1(CCCC)nc(C)c(CC(=O)NC2CC(C(C)NC(=O)C#CC(C)C)C2)s1 CCCC(C(=O)N1CCC(CCC(=O)NCCN(C(C)C)C(C)C)C1)OC CCC(CC(=O)N(CC(C)N(C(=O)CC1(C)CCOCC1)C)C)C(=O)OC Cc1ccc(CCCC(=O)N(C)CC2CCCN(C(=O)CS(C)(=O)=O)C2)cc1 C(=O)(C(C)S(=O)c1ccccc1)N1CC2CC(CN(C(c3ccc(C)cn3)=O)C2)C1 Cc1c(Br)ccc(O)c1C(=O)N(CC(C)N(C(=O)C=CCF)C)C c1(C(=O)NC2CC3(C2)CC3NC(c2cnon2)=O)ccn2ccnc2c1 N(C(=NCCCF)NCc1ccc(F)c(O)c1)C1CCCC(COC)C1 C(=O)(C#CC1CCCOC1)N1CCCC(NC(c2ccc(OC)cn2)=O)CCC1 C1(CC)CCN(C(=O)CSCC(C)C)C1CNC(=O)C=CCN(C)C N1(C(C(=O)N(C)C)=O)CCC2(CC1)CC2(CO)CNC(C1(C)CC2CCC1O2)=O C=CCC(C(=O)N(CC(N1CCC(CC(C)O)CC1)=O)CCOC)C(C)C CC1(C(N2CCC(CCNC(C3CCSCC3)=O)CC2)=O)CC(C#N)C1 C=CCCCC(C(=O)NCCC(F)(F)F)NC(=O)CC1CC2(CCC2)C1 C(C)(C)(CC(=O)NOCC(C)CC)NC(CS(CC)(=O)=O)=O c1(OCCN2C(=O)CCN(CC(C#C)C)C2=O)c(C)nc2c(OC)cccn12 C1(NC(C(CC)=CC)=O)CCN(C(c2nc(CC)ncc2Cl)=O)CC1CO C(=O)(C1=NNC(=O)CC1)N1C(C(=O)Nc2ncccc2[N+](=O)[O-])CC(OC)C1 c1(OC)ccc2[nH]c(=NCC=CCNC(=O)CC3(O)CCCOC3)sc2c1 Cc1ccc(C(=O)N(C(C)CNC(c2coc(C(C)(C)C)n2)=O)C)cc1C(C)C c1(CC(=O)NC(CNC(c2c(CC)csc2)=O)(C)CO)cccc(F)c1O c1(CC(=O)NCCC(C)NC(=O)CN2CCOCC2)csc(C2CCOCC2)n1 C12(NC(C3C4CCC(F)(F)C34)=O)CC3CCC(C1C2)N3C(C1CCOCC1)=O c1(N2CC(CC=C)(N(C(C3(C)CCCN3C(C)=O)=O)C3CC3)C2)ncnc(C)c1F c1(C(N2C(CNC(C3CC4(CC(C)(C)C4)C3)=O)CC2)=O)cnc2c(c1)CCCC2 CC1CC2CN(C(C3C=CCC3)=O)CC2N1C(=O)CCc1cc[nH]n1 O=C(C(CC(F)F)C1CCC1)NC1CCN(C(c2ccnc(O)c2)=O)CC1 c1(C(=O)NC(C2CCOC2)CNC(c2csnc2Cl)=O)c(Cl)n[nH]c1C1CC1 C1(C(=O)NC(C(C)C)CNC(=O)CC2(C)OCCO2)CCCN(C)C1 N1(C(c2ccc(NC)cn2)=O)CCCC(C)(CNC(c2nc(C)n(C)c2C)=O)C1 c1(C(N(C2C3CN(C(c4c(C)nco4)=O)CC32)C)=O)cc(C)c2ccccc2n1 C1(CNC(C(CC)OC)=O)CN(C(C2CCCC(C)C2)=O)CC1C(F)(F)F N1(C(Cc2ccn(CC)n2)=O)CC(F)CC1CC(=O)N(CC(O)COC)C N1(C(C(C)OCC)=O)CCC(CC(C)NC(c2ccnc(CC)c2)=O)CC1 c1(C(C)NCCCCCCC)ccc2c(c1)OC(F)(F)O2 CC1(C#N)CCN(C(=O)C(Cn2cccn2)NC(=O)CC2CCCSC2)C1 Cc1ccc2c(C(=O)NCC(CC(C)C)NC(C3(C)CCCO3)=O)coc2c1 N1(C(CC)=O)CCN(C(c2cccnn2)=O)CC1c1ccc(OC)cc1 C1(CCNC(c2occc2F)=O)CC(F)(F)CN1C(=O)CC1CCCCC1 c1(C(=O)NCC(C)(O)CNC(=O)CC(c2cccc(F)c2)O)ccc(O)nc1Cl CCC(CC)C(F)C(=O)NCC1C=CC(NC(c2c(F)cc(Cl)cc2F)=O)C1 C1(NC(c2cn(CCC=C)nn2)=O)CCCC(NC(c2cnn(C)c2)=O)C1 N1(CC2C(C(C)C)OCCC2)CC(=O)N(CCNCC2CC2)C1=O.c1(S)cccc(F)c1 Cc1nc2ncc(C(N3CCOCC(C(N4CCCCC4)=O)C3)=O)cc2o1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1(NC(CCNC(N)=O)=O)CCC1 CCCC(CCC)CCCC(=O)N1CC2CC(NC(C3CC(=C4CC4)C3)=O)C1C2 C1(CCOC)CN(C(c2ccc(Cl)cc2C)=O)CCN1C(c1cnc(C)nc1)=O N1(C(=O)C=Cc2ccoc2)CCOC2(C1)CN(C(c1ccc3c(c1)OCO3)=O)C2 C1(C(=O)NCC2C(c3ccn(C)n3)C2)CCN(C(=O)CO)CCC1CO C(N=c1ccnc(NCCSc2n[nH]c3c2CCCC3)[nH]1)c1n(C)nc(C2CC2)c1 N1(C(=O)OCCCCC)CC2C=CC1C(C(=O)N(CCCCOC)C)C2 c1(Cn2c(C(C3CCCO3)C)nc(-c3cncnc3)n2)nc2ccccc2o1 c1(C(=O)NCC(C)NC(c2cc(OCC)n[nH]2)=O)cc(O)ncc1Br N1(C(C2CCN(C)C2)=O)CC(NC(=O)CCCc2cccc(Cl)n2)CC2(CC2)C1 c1(OC)coc(C(=O)NC(CNC(C2CCCS2)=O)C(C)C(C)C)cc1=O C1(OC)CNC(=O)C1.C1(N(C)C)CCC(Cn2cc(C3C4COCC34)nn2)CC1 CC1c2c[nH]nc2CCC1C(=O)N(C)CC1CN(C(c2cc(Cl)nc(Cl)c2)=O)C1 C1(=CC(=O)NCCC2(OC)CN(C(C(CCSC)OC)=O)C2)CCCCC1(C)C c1(CNC(N(CCCN(CC)CC)C)=O)ccccc1-n1cncn1 C(=O)(CCC(F)(F)F)NC(CNC(C(C)NS(C)(=O)=O)=O)(C)C1CC1 C1(OC)CCC2(C(=O)NC(C(=O)NC3(C)CCSCC3)C(C)C)CC12 C1(C(=O)NCCN(C(c2n(C(C)C)ncc2)=O)C)CN2CCCC1CC2 C1(NC(C(F)=CC)=O)CCN(C(c2ccccc2)C(=O)NC)CC1O CC(C(=O)NCC(C1CC1)NC(=O)CNC(c1nccs1)=O)n1ccnc1 N1(C(C(C)=C2CCC2)=O)CCCC(C2CC2NC(C2CC3C=CC2C3)=O)C1 N1(C(c2ccc(C)cc2)=O)CCCC2(NC(c3ccc(C)cc3F)=O)CCCC12 Cc1cc(C(N2CCOCC2CN(C)C(C2(C(F)F)CCCC2)=O)=O)c(C)s1 CC1=CCSC1C(N1C(C(N2CC(F)(CO)C2)=O)CC1C)=O C12CC(=CC1O)C(=O)N2CC.C(=O)(CCC(=O)N1CCOCC1)NCCC(N)=O C1(C(=O)NCC(C(C)C)NC(C2CN(C(C)C)C2)=O)CCOC(C)(C)C1 c1(NCC2CC(C)OCC2)ncc(F)cc1N C1(COC)CCC(C(=O)NC2CC2c2ccoc2)O1.C12(CC(CO)C1)C(=O)N2 C(C(C)(O)C(C)(C)C)NC(C(CNC(=O)C(N1CCOCC1)C)OC)=O CONC(=O)C(=O)N.c1(C2CC(=O)c3cc([nH]n3)C=CCN2)cccc(C)c1 c1(OC)ccc(NC(C2CC2CNCc2ccc(N(C)C)cc2)=O)c(C)c1C Cc1nccc(C(N2CCC(O)(CN(C)C(c3cn(C)nc3Cl)=O)C2)=O)n1 c1(C(N2CCC(NC(Cc3nnc(C)o3)=O)C(C)C2)=O)cc(C#N)c(N)cc1O C1(C(N2C(CNC(CC3CC(OCC)C3)=O)CCC2)=O)CCC(C)C(C)C1 N1(c2nnc(-c3cccc(OC)n3)n2CC2CCCO2)CCn2nnc(Br)c2C1 c1(C(=O)NCCN(CCC)C(c2ccc(C(C)C)nc2C)=O)ccc(O)cc1F c1(CC(C(=O)N2CCC(c3cnn[nH]3)C2)NC(C2(CC)CC2)=O)cnn(C)c1O O=C(O)CC1CCN(Cc2cccc3sccc23)c2ccccc21 Cc1nnccc1CNC(=O)CCN(C(=O)C(C)(C)C1CCCO1)C(C)C N1(C(CCC#CC)=O)CCN(C)C(CNC(c2cccnn2)=O)C1 c1(C(=O)NC2CCCC2NC(c2cnc(O)o2)=O)ccc2c(c1)CCC=C2 CCCC(C)(CC)C(=O)NCC1COCC1NC(c1cnc2sccn12)=O N1(CC(N2C(CC)C(NC(=O)C(O)c3cnc[nH]3)CC2)=O)C(=O)C(=O)N(C)C1=O C1(NC(C(CSC)OC)=O)CCN(C(c2csc(C(F)F)c2)=O)CC12CCC2 C1(C(=O)NCC2(OCC)CN(C(C3CC3CC)=O)C2)Cc2cc(C)ccc2O1 C1(NC(=O)Cc2ccc(Br)nc2)CC2(C1)CN(C(=O)Cc1cccc(F)c1)C2 C1(C(N(CCN(C(C)C)C(C2CCOCC2(C)C)=O)C)=O)CC2(C1)CC1(CC1)C2 CC(CC(=O)NCC(C)NC(=O)C(CN(C)C)c1ccccc1)C(C)(C)C Cc1cc(C#N)cc(CNC2CCCN2)n1.C12CCN(CC1)CC2 C(=O)(C(C)(C)C1=CCSCC1)NCC1(C)CCN(C(c2c(C(C)C)ccs2)=O)C1 C1(CC(N2CC(F)(CNC(C(C=CC)O)=O)C2)=O)CCCS(=O)(=O)C1 c1(C(CC(=O)OC)NC(=O)NC2CCCN(C)C2)ccc(O)c(C(C)(C)C)c1 C(=O)(C1=COc2ccccc2O1)N1CCN(C(c2cnn(C)c2N)=O)C2C1C2 C(CCS(=O)(=O)c1ccccc1)NC(c1cc(C)n(C2CCOC2)c1C)=O N1(C(c2cc(CC)on2)=O)C2CCC1C(CNC(=O)CSCc1csc(=N)[nH]1)C2 N1(C(C(C(C)C)F)=O)CCC(C2(NC(c3ccc4ncnn4n3)=O)CC2)C1 c1(OC)ccc(NC(=O)C(=O)NCC(C)(C)N2CCCC2)c(C)c1OC N1(C(C2CN(C(C)C)C2)=O)CCCN(C(c2ccc(Cl)[nH]2)=O)C(C)C1 c1(CCC)ccccc1C(=O)NCCOCCCN(C)C(C1CCSC(C)C1)=O N1(C(c2c(CC)nc(C)[nH]2)=O)CCCC(O)(CCNC(=O)C=Cc2cc[nH]c2)C1 N1(C(C=C(C)c2ccsc2)=O)CCN(C(c2c(N)sc3c2CCC3)=O)CCC1C CCC(C)(C)C(O)C(=O)N1CCCCC1CN(C)C(c1nc(Br)c[nH]1)=O C(N=c1cc(C(=O)N(C)C)nc(Cl)[nH]1)C1CCN(C(C2(C)CCCC2)=O)C1 N1(C(C2N(Cc3cnc(CC)s3)CC(F)(F)C2)=O)CC(C)OC(C)(C)C1 c1(C(=O)NC(C(C)NC(=O)Cc2ccnc(Cl)c2)C)ccc2ncc(Br)n2c1 C(=O)(CCCCCCCCCOC(C)=O)NC(C1CCC(=C)CC1)(C)C Cc1nc(CO)ncc1N.C1(CC(C(=O)CCC2(N)CCC2)=O)CCOC1C C(c1ccc(C(N)=O)o1)=CC(=O)N(C(C)CN(C(=O)C(c1ccccc1)F)C)CC C1(NC(=O)CC2CCCC2)CC(O)CN(C(=O)CCc2ccccn2)C1 c1(CC)nc(C)oc1C(=O)NCCn1ccc(C(=O)N(CCCF)CC)c1 C=CC(C)CCN=c1nc(N(C)Cc2ccc(C3CC3)cn2)c2c([nH]1)CCS2 CC1(NC(=O)Cc2cccc(Cl)c2)CCN(C(=O)COC2CCOCC2)C1 c1(C(=O)NC2CCC(C(=O)NCC(=C)C)C2)ccc(OC)nc1 C1(OC)CN(C(=O)CCc2ccc(Cl)s2)C(C)(CNC(=O)C2=CCC2)C1 C1(N(C(C2C(C(C)C)C2)=O)C)CCN(C(C23CC(CO2)C3)=O)CC1 N1(C(COCCCC)=O)CCN(C(=O)CC2(C#N)CC2)C(CCNC(=O)NC)C1 C#Cc1cnc(C(=O)NC(CO)C(C)NC(c2cccc(C=C)c2)=O)c(C)c1 c1(C(=O)NC(C(C)C)CCN(C(=O)CCF)C)nc(Cl)ccc1N N1(C(C(C)N(C(=O)OC)C2CC2)=O)CCOCC1CC(=O)NCC(C)C1CCC1 N1(C(COC(CC)C)=O)CCCC(C2CN(C(c3cc(I)c(F)cc3F)=O)C2)C1 N1(C(C2(CSC)CC2)=O)C2CN(C(=O)C(CN(C)C)c3ccccc3)CC12 Cc1ccc(C(=O)N(C2CCCC(N(C)C(c3nc(C)oc3C)=O)C2)C)c(O)c1 C1(C(=O)OC)CCN(Cc2ccc(CCC#N)cc2)C2CCCC12 C1(CCC=C)(NC(=O)CC2C=CCCC2)CN(C(=O)CCOC2CCC2)C1 Nc1ccc2nc(NCC3(F)CCCN(C(C4(CO)COC4)=O)C3)sc2c1 C1(CCNC(=O)CSc2n[nH]c(C)n2)(OC)CN(C(=O)Cc2cnns2)C1 C12(C(=O)NCC(C)(C)NC(c3cc(C)c(C)s3)=O)CCCCN1CCC2 CCCCC(CC)CC(=O)NCC1(C)CC(F)(F)CN1C(=O)CC(=O)NCC c1(C(N2CCC(Cn3cc(C(CC)O)nn3)C2)=O)cc(C)cc(C#N)c1 C1(C2CCCC2)(C(=O)NCC2N(C(c3c(C)cns3)=O)CCCC2)CCNC1=O C(N=c1[nH]n(C)c2c1CN(S(C)(=O)=O)CC2)c1cccc(C)c1Br C=C1CC2(C1)CC(C(N1CC3(CNc4cc(=O)c(OC)c[nH]4)CC1CO3)=O)C2 c1(OCC(=O)NCC(N2CCS(=O)CC2)=O)ccc2c(c1)CCC2 C=C1CCN(C(=O)CC2CCCN2C)CC1C(=O)NCC(C)C#N N#Cc1cc2cc(C(=O)NCC(F)CNC(=O)CN3CCC(O)CC3)[nH]c2cn1 C(=O)(C(C)(C)C(F)F)NCCC1CCN(C(COCc2nnc(C)s2)=O)C1 N1(C(CC=C)=O)CC2(CCC2NC(=O)CCOc2cccc(C(C)(C)C)c2)C1 c1(CC)ccccc1C(N1CCCC1C(C)NC(c1ccsc1C)=O)=O.C(C(N)=O)S C1(CC#C)(C(=O)NCCC2CCOCC2)CCN(C(=O)CCC2CCCCO2)C1 c1(C(N(CC(CC)NC(CCC#CC)=O)C)=O)nccc(Cl)c1C C1(C)(NC(c2cc(CC)sn2)=O)CCCCC1C(=O)NCc1ncc(C)[nH]1 N1(C(C2CN(C(=O)NC)C2)=O)C2CCC1CN(C(C1CC(SC)C1)=O)C2 c1(CC(=O)NCC2CC3CCC2CC3)c(Cl)cccc1B(O)O c1(C(=O)NCC2(NC(CSC)=O)CCCCC2C)ccc2c(c1)OCO2 C1(CC(=O)N(C(CC)CC)CCO)CC2CCC1CC2 c1(C(C(=O)N(CC(CCC)NC(=O)C=Cc2cn(C)nn2)CC)C)ccc(F)cn1 O=S(=O)(c1ccc(N2CCSC(CO)C2)cc1Br)N1Cc2ccc(Br)cc2C1 C(C(C)(C(N)=O)NC(C1CCCN1C(=O)CC12COCC(C1)C2)(C)C)OC c1(NC(=O)COC=CC(N2CCC(SCC)CC2)=O)cc(C)ccc1C(C)C CCCC(C(=O)NC12CC(CNC(c3ncc(Cl)nc3Cl)=O)(C1)C2)C(C)C N1(C(C=C(C)C)=O)CCC2(CC1)CC2C(=O)NCCn1ncccc1=O C1(C(=O)NCC2=CCN(C(c3cn(C)nc3Cl)=O)CC2)COc2ccccc2O1 C(C(=O)NC1CC(NC(C2CNC(=O)N2)=O)C1)(C(C)(C)C)c1ccc(C)cc1 N1(C(C(CCN(C)C)O)=O)CC(C(=O)NC2CC(OC(C)(C)C)C2)C(C2CC2)C1 c1(NC(c2c(Cl)ccc(Br)c2F)=O)cc2ccccc2c(Cl)n1.C12CN(C1)C2=O C12(C(=O)NCc3cccc(NC(c4c(C)con4)=O)c3)CCC(C)(CO1)C2 C1(NC(CN(CCOC)C)=O)CN(C(c2ccc(N)c(O)c2)=O)CCC1CO Cc1ccc(C2(O)CN(C(c3ccnn3C3CC3(F)F)=O)C2)cc1 c1(C(=O)NC(CNC(c2cncc(OC)n2)=O)C2CC2)cn2c(n1)SCC2 Cn1cc(S(C)(=O)=O)c(C(=O)NC2CCC2NC(=O)CCCC2OCCO2)n1 Nc1cc(C(N2CC3CC(NC(=O)CC4CCC45CCC5)C2C3)=O)cc(O)c1Cl C1(NC(c2ccc(C)nc2O)=O)CC2(CCN(C(c3cnc(O)cc3C)=O)C2)C1 C1(CCOC)CN(C(=O)C(COC)COC)CCN1C(=O)CCNC(C1CCC1)=O c1(C2N(C(C3CCN(C(c4nc(CC)oc4)=O)C3)=O)CCC2)ccc(O)cc1 CC1(C)COC(CC(=O)NC2(CO)CN(C(C3CC4CCCC4C3)=O)C2)CO1 CCC(C)C(=O)N1CC(NC(=O)CCc2nncn2C)C1 c1(C(=O)NCC(C2CCC2)NC(C(C)OCC(C)C)=O)ccc(=O)n2c1CCC2 CCCCCCCCC(F)C(=O)NCC1CC1CNC(=O)C(C)NC(=O)NCC CCC(C)(C)CC(=O)NC(C)(C)C(=O)NCC1CC1NC(N)=O Cc1nc(C(C)NC(C2CC(NC(c3cc(Cl)no3)=O)CCO2)=O)c(C)o1 C(=O)(C#CC(C)(C)C)N(CCC(C)NC(c1c(OC)noc1C)=O)C C1(C(N2C(C(=O)NCCCc3ccccc3)COCC2)=O)CCC2(CC1)CC2 C(c1ccccc1)=CC(=O)NCC(c1ccccc1)NC(=O)C(F)n1cccn1 c1(CC(=O)NCCOCCC(=O)NCC(O)C(F)(F)F)ccccc1F c1(C(=O)NCC2N(C(c3cc(CC)cc(C)c3)=O)CC2)cc(C)c(F)cc1N C1(NC(C(C)SCCCC)=O)CCN(C(c2sc(CC)nc2C)=O)C1(C)C c1(OCC)ncccc1C(N1CC=CC1CNC(=O)CN(C1CCCC1)C)=O N1(C(C2(CCCl)CC2)=O)CCC(O)(c2cn(-c3ccc(Cl)cc3F)nn2)CC1 C12(C(N3CCC(C)(NC(Cc4c(C)occ4)=O)C3)=O)CCC(F)(CC1)C2 c1(C(N2CCCC(CNC(COCCCCC)=O)C2)=O)ccn2ccccc12 C(=O)(C1=C(F)CN(C(=O)C(C)CC2CCCC2)CC1)NCc1cncc(C)c1 C1(CNC(=O)CN2CCCCCC2)CCCCN(C(C2CCCS2)=O)C1 C1(C#N)(CNC(CCC(C)NC(c2cc(=N)[nH][nH]2)=O)=O)CCOCC1 c1(NC)cc(Cl)ccc1C(N1CCC(O)(CNC(C2CCC2(F)F)=O)C1)=O c1(CC)cc(C(=O)NC(Cc2ccoc2)C(=O)NCC(N2CCOCC2)C)cs1 N1(C(c2c(C)cccc2)=O)CC2CN(C(c3ccoc3I)=O)CC12 c1(CN2C(CN3CCC(N4C(=O)CCC4)CC3)CCC2)nc2cccc(F)c2[nH]1 N1(C(c2c(C)nc[nH]2)=O)CCC(CNC(c2ccc(=O)n(O)c2)=O)C1(C)C CC(C)(C)CCCCC(=O)NC1(C)CCN(C(=O)CC2CCCCC2O)C1 c1(C(N(CCCN(C)C)CCN(C)C)=O)ccc2c(c1)C(C)(C)C(=O)N2C c1(C(N(C)CC2(F)CCC(C(=O)O)CC2)=O)cccc([Si](C)(C)C)c1 N1(C(C(=O)NCCOC)=O)CCC(N=c2cc[nH]cc2C#N)CC(C)(C)C1 C(CC(C)CC)(C(=O)N1CC=CCC1)N(C(C1CC(CCC)C1)=O)CC Fc1cc2nc(N3CCOCC3)cc(NCCc3cc(F)c(Br)cc3F)c2cc1F N1(Cc2c(C)n[nH]c2)CCC2(CC1)CC(C(=O)Nc1nccc(Cl)c1I)CO2 c1(NC(=O)Nc2c(C(C)C)c[nH]n2)cc(C(F)(F)F)cc(Cl)n1 c12ccccc1C2.C1(NC(C(=O)N(C)C)=O)CCCC1C(=O)NC12CCC(C1)C2 n1(C(C)C)ccc(C(N2CCC(CNC(c3cnn(C4CC4(F)F)c3)=O)C2)=O)n1 N1(C(C2N(C(C3CCN(C)C3)=O)CCC2)=O)CC(CO)CC12CCC2 Cc1cc(O)ccc1NC(C1CC=CCN1C(C1CCCS1)=O)=O N1(C(C(=O)NC2C(=C)CC2)C2CC2CSCC)CCCN(C(=O)OC(C)(C)C)CC1 N(C1CCCc2c(CBr)cccc21)C(C1(NC)CCN(CCNS(C)(=O)=O)CC1)=O C(C(=O)NCc1nccnc1C)(C(C)(C)O)NC(c1cc(OC)n(C)n1)=O c1(NCCOCC=C)[nH]c(=NCc2nccn2C(C)(C)C)nc2scnc12 c1(CC)cc(COC(=O)CC2CCCOCC2)ccc1F CCCC(C(=O)NCC1(C(N)=O)CN(C(c2ccnnc2S)=O)C1)C(C)C C(=O)(CC1=CCN(C)CC1)N1CCCC(N(C(c2nn(C)c(Cl)c2Cl)=O)CC)C1 CC1(C)C=CC(N=c2nc(N3CCC(N4CCC4)CC3)c3ccccc3[nH]2)CC1 C1(CC(=O)NC(C2(CNC(c3ncccn3)=O)CC2)C)CCCCC1O c1(C(=O)NC2CC(CNC(CNS(C)(=O)=O)=O)C2)cnn(C)c1C(F)F Cc1ccc(C(N2CC3(CC(CNC(=O)CSc4n[nH]c(O)n4)C3)C2)=O)c(C)c1 C#Cc1ccc(C(N2CCCC(CCCCNC(=O)CS(=O)CC)C2)=O)cc1F C1(NC(C(C)OCC)=O)CCN(C(c2ncc(Cl)nc2Cl)=O)CC1C O=C(CCOCCCNC(c1cnsc1)=O)NCCn1cnnc1 C1(C(N(CC(CCC=C)O)C)=O)CC2CCC(C1)N2C(=O)C(C)C(F)F C1(N(C(c2c(OC)ccs2)=O)C)CCN(C(C2CCC(O)CC2)=O)CC12CC2 c1(C(=O)NC2CCCN(C(CCCOCC)=O)C2)ccc2c(c1)C1CCC2O1 C=CCC(C(=O)NC1CN(C(=O)CS(=O)(=O)NC)CC1O)C(C)C N1(C(C2(NC(c3ccc(O)cc3)=O)CCN(C)C2)=O)CC2CCCCC12 c1(OC)cc(C(=O)NCC2CCN(Cc3cccs3)CC2)ncn1 c1(OC)ccccc1C(CNC(=O)C(C)CF)NC(=O)C(O)C1CCCC1 c12cccc(c1)NC(=O)CCc1nnc-2o1.c1(COCC)ccsc1Cl c1(C(=O)NCC2(COC)CCN(C(=O)C(C)SC)C2)ccnc(C)c1C c1(OC(C)CNS(=O)(=O)CCCO)ccc(Br)cc1 C1(O)(CNC(c2c(CCC)n[nH]c2)=O)CC2CCC(C1)N2C(=O)Cn1nccn1 c1(CC(=O)N(CCC)CCC)ccc2cc(OC)ccc2c1 c1(CC(=O)Nc2ccnc(F)c2F)n[nH]c2ccc(-c3ccc(F)cc3F)cc12 c12ccc3[nH]c(cc3c1)C(=O)NCCCNC2=O.c1(OC)cccc(CO)c1.C1(C)CC1 Cc1ccc(F)c(CNC(C(C)(C)C)c2nnnn2CC(F)F)n1 CS(=O)(=O)CCCCS(=O)(=O)N1CCCCCC1c1noc(-c2ccccc2)n1 c1(CC(=O)NC2CC3N(C(CCSC)=O)C(COC3)C2)coc2ccc(F)cc12 Cc1ccc(CNC(=O)C(=O)NCc2cnn(C(F)F)c2)cc1C#N C1(O)(CC(=O)NCCCCN(C(C2CC(CCC)C2)=O)C)CCCOC1 Cc1cc(F)c(Cl)cc1C(=O)NC(C)C(CO)NC(c1cccc(CO)n1)=O c1(NC(=O)NCC2C(C)(C)C3CCC2C3)ncn2cc(Br)cnc12 Cc1ccc2[nH]cc(CC(=O)NC(C(C)NC(=O)C(C)C(C)C)C(C)C)c2c1 c1(NC(C(COC)OC)=O)cnc2[nH]cnc2c1.C12CCC1C(=O)NC2 Cn1nc(C(N2CCCC(NC(c3c[nH]nc3C(C)(F)F)=O)C2)=O)cc1CO n1(CC)nc(C)c(C(N2CCC(C(C)NC(c3nc(Cl)sc3Cl)=O)C2)=O)c1Cl c1(CC(=O)N(CC(C)NC(=O)C#CC2CC2)C)cc(Br)c2c(c1)CCO2 C=C=CC(C)C(=O)N1CCCC(CC(N2CCC(O)(COC)C2)=O)C1 C1(F)(C(N(CCNC(C(CC)Sc2ccccc2)=O)CCOC)=O)CC=CCC1 C1(NC(C2(CCN(C)C)CC2)=O)CC(C(=O)N2CC3(CC(F)C3)C2)=CC1O C1(C(=O)NCC2CC(C)N(C(=O)CC3(O)CCCCC3)C2)CC2(CCC2)CO1 CN1CCCC(NC(c2csc(CNC(=O)C=CC3CCCCC3)c2)=O)C1 C(=O)(C1=CCCCC1)NCCNC(CC(c1ccc(C(C)C)cc1)C)=O c1(C(N2C3(CNC(C(CC)(F)F)=O)CC(C2)C3)=O)cc(C)n(-c2nccs2)c1C CCCC(C(=O)NCC1(O)CC(NC(c2cc(C)c(C)s2)=O)C1)OCC N1(CC=CC(=O)NC(C)CNC(=O)C=CC(C)(C)C)CCCCC1 C(CCCCCC(=O)N(C(C)CNC(c1ccc(Cl)c(Cl)c1)=O)C)SC C#Cc1ccc(C(=O)NC2CC2NC(c2ccccc2OCCCC)=O)cc1C N1(C(c2cc(OCC)n[nH]2)=O)CCC2CCCC12C(N1CC(C(N)=O)C(C)C1)=O C1(NC(CC2(OC)CCC2)=O)C(C)CCN(C(c2ccc(C)c(N)c2)=O)C1C C1(CNC(CN2CC(C)C2)=O)CC2CCC(C1)N2C(c1ccc2[nH]ccc2n1)=O C1(NC(CC2ON=C(C)C2)=O)CCCCCC1C N1(C(CNC(=O)CC2CCCCC2)=O)CCC2CCCC12CC1CCCNC1=O C(C(C)CC(=O)NC1CC(CNC(=O)C(C)NCC(C)C)C1)OC C1(C(=O)NCC2CN(C(C)C)C2)CN(C(C2CCS2(=O)=O)=O)CCO1 CC(=O)CCCC(C)C(=O)NC(CCC(=O)Nc1cc(C)cc(C)c1O)C(C)C C1(C)(CC2(CC(C)(C)C)N=N2)COCCN1 CC(C)CC(F)C(=O)NCC1CC1CNC(=O)CCc1ccc(Br)cc1F c1(C(C)C)ccncc1NC(=O)CCN(C(=O)C(C)NC(N)=O)C C1(C(N(CCOCCCOC)C)=O)CC(NC(C2(C)C(C(=O)OC)C2)=O)C1.C1CC1 C=CCCCCCCNC(=O)C(C(C)(C)O)NC(=O)CNC(=O)C(C)CC N1(C(c2c(OC)ccc(C)n2)=O)CC2CC(C1)N(C(=O)Cc1cnn(C)c1C)C2 N1(C(c2ccc(CC)s2)=O)CCC2CN(C(=O)Cc3ccccc3)CCC12 N1(C(Cc2ccc(C(N)=O)cc2)=O)CC2(CCC2CNC(=O)Cc2ccns2)C1 CC1CC(C(=O)Nc2cccc(NC(C3(NC(N)=O)CCCC3)=O)c2)CCO1 N1(C(Cc2cccc(OC)c2)=O)CCN(C(=O)C2=NOC(C)C2C)CC12CCC2 C(=O)(C(CNC(C1CC12CC2)=O)C(C)C)NCC1N(CC)CCCC1 CCCCCCS(=O)(=O)N1CCC(CC(=O)Nc2ccc(N(C)C)cn2)CC1 C(=O)(C(Cc1cnc[nH]1)NC(c1scnc1C)=O)NC1(CC=C)CCC1 C1(CNC(CN(CC(C)C)C(c2n(CC)ccn2)=O)=O)COCC(=O)N1C c1(C(=O)NCC2CCN(C(C#CC(C)C)=O)CC2C)cc2c(cc1Cl)NCC2 C(=O)(C1=CCCC1)NCC1(CN(C)C(C2CC3(C2)CC3F)=O)CC1 C1(C(N2C(CNC(C(C)SCc3ccccc3)=O)CC2)=O)CCCC(C)(C)O1 N1(C(CC(C)C(F)F)=O)CCCCCC(NC(=O)C=C2CC3CCC(C2)N3C)C1 C(=O)(CC1=CCOCC1)NC(CCCOC)C(=O)NCC(F)Br N1(C(C(C(C)C)N(C)C)=O)CCC2(CC1)CC(C)N(C(=O)C(O)C1CCC1)C2 CC(C)CCCCC(=O)N1CC(C)(NC(=O)C2=C(C#N)CCC2)C1 Cc1cc(N)ccc1C(=O)NC1CCCC(NC(=O)Cc2nncn2C(C)C)C1 CP(C)(=O)C1CCC(NC(=O)NCCCNc2ccccc2)C1 CN1CCCC1C1CCCCN1C(c1cc(F)ccc1C(F)F)=O c1(C(=O)NCCCCNC(C2C(=C)C2)=O)ccc2c(c1)OC(C)(C)C2 Cc1cc(CC(=O)NC2(C(=O)NC3CCCC3n3cccn3)CCCC2)cs1 c1(OC)ccc(Br)cc1C(N1CC2CN(Cc3ccccc3N(C)C)C2C1)=O.NCC C1(CNC(C(CCOC)C)=O)COCCN(C(=O)CNC(=O)CC2(C)CCCC2)C1 C1(CC(=O)NCC2(COC)CCC2)CCN(C(c2cc(C)cc(C)c2)=O)C1(C)C CCCCC(O)C(C)C(=O)N1CCC(CCNC(c2cccc(N)c2C)=O)C1 C(C(C)C(=O)NCc1ocnc1C(=O)NCC1CCC=CO1)OC Cc1cc(C(N2CCC(C(C)NC(=O)COCC(F)F)C2)=O)c(F)cc1Cl C#Cc1ccc(C(=O)NCCC(C)NC(=O)C(C2CCCCCC2)C)c(F)c1Cl N1(C(CCCCNC(C)=O)=O)CCCC12CCN(C(C1C(C(F)F)C1(F)F)=O)C2 c1(C(N(C2CCCCN(C(C(CC#C)C)=O)C2)C)=O)cc([N+](=O)[O-])cnc1O C1(O)(C(N(C)CC2CCCN(C(C34CCC(CC3)C4)=O)C2)=O)CC2CCC1C2 c1(OC)cc(Cl)cc(C(=O)NCC(N2C(C(=O)OC3CC3(F)F)CSC2)=O)n1 C1(NC(c2cnc(OC)nc2C)=O)C(C)CN(C(c2ccc(N)cn2)=O)CC1C N1(C(c2scc(C)c2)=O)CCC2(CNC(=O)CCCC(F)(F)F)CCCCC12 C(=O)(CS(=O)(=O)NCC1CCCO1)NC1C(NC(CCOC(C)C)=O)COC1 C#CCC(C)(CNC(C1COCC1NC(=O)Cn1ccnc1C)=O)CO Cc1ccc(S(=O)(=O)n2ccc(C(=O)N(CC(C)NC(=O)C(C)(C)C)C)c2)cc1 N1(C(c2cccc(C(F)(F)F)c2F)C(=O)NC)CCCC2CCNC(=O)C12 N1(C(CCN(C)C)=O)CCC(CC(=O)NC2(c3ncc[nH]3)CC2)C1 c1(CC)n[nH]c(CC)c1CC(=O)NCc1cn(CC(C)NC(=O)C(N)=O)nn1 C1(C2CC2)(C(=O)NCC=CC(=O)NCC(C)(C)O)CC(=O)C1 c1(C(=O)NC2C(NC(CC(C)C3CCCC3)=O)CC2)c[nH]c2ncccc12 Cc1c(C(=O)NCCC2(O)CCN(C(C3CC(O)CN3C)=O)C2)cccc1F C12(CNC(c3c(C(C)C)scn3)=O)CCCCC1N(C(=O)C=CS(C)=O)CCC2 c1(C(=O)NCCN(CCC)C(c2nocc2Cl)=O)cc(C(C)C)on1 N1(C(c2ccc(CC)s2)=O)CCC2C(C1)NC(=O)CN2C(=O)CC(C)N(C)C N1(C(=O)NC(CC)(C)C)CC2(CC(NC(C3CC3(c3ccc(C)o3)CO)=O)C2)C1 Cc1c(N(C2CCN(C(=O)C3=NNC(=O)CC3)C2)C)nc(C2CC2)nc1Cl C1(CNC(C(C)OCCC=C)=O)C2CCC(C2)N1C(=O)CC=CC(C)(C)C C=C(C)C(C)(C)C(=O)N1CC(NC(c2cc(C)n(C(C)C)n2)=O)C1 c1(C(N(CCNC(CC2CCCC(C)C2)=O)C)=O)cnc2c(n1)CCCC2 Cc1cc(NC(c2nnnn2CC)C2CC23CCC3)ccc1OC(F)F.C(C)(C)C CC1CN(C(=O)C(F)C(C)(C)O)C(C)CN1C(=O)Cc1ccoc1 Cc1cccn2cc(CC(N3CCCC4(NC(=O)CSC(F)F)CC4C3)=O)nc12 N1(C(=O)Cc2ccnc(Br)c2)CCN(Cc2ccccc2)C2CCCCC2C1 N1(C(CCCC(CC)NC(=O)C(CC)SC)=O)CCc2cccc(O)c21 C1(CNC(CC=C=C)=O)CC2CCC1N2C(c1cnn(Cc2ccccc2)n1)=O N1(C(CC(C)OC)=O)CC(C2CC2)(C(=O)NCC(C2CC2)C2CC2)C1 c1(C(N2C(CCNC(C=CC=CCC)=O)CC(F)(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(C(=O)NC2CC(CNC(CCc3n(C)ccn3)=O)C2)cccc(C(C)(F)F)c1 c1(CC(c2ccccc2)CNC(=O)NCc2ncc(C)cn2)ccc(Br)cc1F CC1(C)CN(CCC(=O)N2CCC2CNC(=O)C=C(Cl)Cl)CCS1 c1(C(=O)NCCCCC(C)NC(c2ccccc2Cl)=O)cn(C)c(=O)cn1 C1(C(=O)NC2C(C)CN(C(=O)CCSCC(N)=O)C2)CC12CCC(C)(C)CC2 C1(CNC(CN(c2ccccc2)CC)=O)(CO)CCN(C(=O)C#N)CC1 c1(C(CSc2cc(C(=O)O)no2)NC(Cn2ccc(C)n2)C)ccc(O)cc1 C1(C(C(=O)NCCCF)N(C)CC2CCCC23CC3)CC2CC1C1CC21 C1(C2CCCN(C(=O)C3CC3)C2)(NC(C(c2ccc(C)cc2)C)=O)CC1 N1(C(C(CCSC)(C)C)=O)CCC(O)C(N(C(=O)CS(C)(=O)=O)C)C1 c1(C(C)NC(COC)=O)ccc(S(=O)(=O)NC2CC2)s1 n1(CC(=O)O)cnc2ccccc12.CN1CCC(C(=O)NOCCF)C1 C1(C(N2C3CC(NC(=O)CN4CCSCC4)(C3)C2)=O)CC2C=CC1C21CC1 C1(NC(CN(C(C(CCOC)OC)=O)C2CCC2)=O)CC12CCCCC2 CC(CC(=O)N(C1CCCN1C(=O)CC(Cl)Cl)C)n1ccnc1 c1(C(=O)OC(CC)CC)cncn1-c1cnn(C)c1 C1(O)(CCNC(COCC=C)=O)CCN(C(=O)Cc2ccccn2)C1 C1(NC(C2CC(N(C)C)C2)=O)C(C(=O)NCCC2(COC)CC2)CCC12CCC2 C(=O)(C1=CC(C)(C)C1)NC(=O)CN1CCCC(n2cc(CSCC)nn2)C1 C1(NC(c2ncc(C)nc2)=O)CN(C(=O)CCCC2CCCO2)CC1C1CC1 c1(C(C)C)nc(CC(=O)NC2CCC2CNC(=O)CC2(C)OCCO2)cs1 C1(N(C)C(c2sccc2-n2cnnn2)=O)CN(C(c2ncc(F)cn2)=O)CC1F N1(C(C(c2ccc(F)cc2F)C)=O)CCOC2(CCN(C(=O)CN=S(C)(C)=O)C2)C1 C(C(C)(O)C(=O)NCC(C)CN(C)C(c1ccc(Cl)cc1)=O)OC c1(NCC2(O)CN(C(C3C(=C)CC3)=O)C2)ncnc2c(Br)nn(C)c12 C1(O)(CCNC(C2(CC(C)C)CCC2)=O)CCN(C(C2CCC(=O)N2C)=O)C1 S(=O)(=O)(CCCCCCl)N1CCC(C#N)(NC(COC(C)C)=O)C1 CONC(=O)C(=O)N1CCC(c2ccccc2)(NC(=O)C(C)N(C)C)C1 Cc1nccnc1C(N1CCCC(N(C(c2ccc(Cl)s2)=O)CC2CC2)C1)=O c1(C(N(C2CCN(C(C(C(C)C)SCC)=O)CC2)C)=O)ccnc(Cl)c1O C1(NC(CCNS(C)(=O)=O)=O)CN(C(C2CC3(C2)CC32CC2)=O)C2(CCCC2)C1 c1(C2C3(O)CC(C3)N2)nnnn1C(C)C.C(C(C)(C)OC)OCC n1(CCCC)ncc(C(N2CC(NC(c3cc(C4CC4)ns3)=O)C(C)C2)=O)c1C c1(-c2scc(C(=O)Nc3cc(OC)c(F)cc3Br)n2)ccc2cnn(C)c2c1 C12(SCCOCCN(C(CN(C(C)C)C)=O)C)CCC(CC1)CO2 N1(C(N2CCCC2CN2CCCC2)=O)CCCCC2(CCOCC2)C1 C=CC1CN(C(=O)C(O)COC)CC1NC(=O)CCc1ccc(OC)c(Cl)c1 C(=O)(C#CC1CCOC1)NC(c1ccc(C)cc1)CNC(=O)Cc1nc[nH]n1 N1(C(C2CC3CC(OC)C3C2)=O)CCCC12CCN(C(=O)C(Cl)=CCl)CC2 N1(C(c2ccnc(O)c2)=O)CCC(N=c2c(Cl)c[nH]cc2[N+](=O)[O-])C1 c1(CC)ccccc1C(=O)N(CCCC(=O)NC(c1ccco1)C)C(C)C C1(C(=O)NCC2(NC(C3CC4(C(OC)CC4)C3)=O)CCC2)CC(C)(C)CCO1 N1(C(C(c2c(C)nn(C)c2C)C)=O)CC2CN(C(=O)C3=NNC(=O)C3)CC2C1 C1(C(=O)NC2C(CN(C)C)CCC2)C2CCN(C(C3(F)CCCC3)=O)CC12 Cc1ccc2[nH]cc(C(=O)NC3CCN(CCn4ccnn4)CC(C)(C)C3)c2c1 CC(CC(=O)N1CC(NC(=O)C(O)Cc2cnc[nH]2)C2(CC2)C1)P(C)(C)=O c1(C(N2CCCC(C(C)NC(c3ccc(C#C)o3)=O)C2)=O)c(C)cc(C)cc1C N1(C(c2c(CC)nc(C)[nH]2)=O)CCC(NC(c2c(C)cc[nH]c2=N)=O)C(F)C1 Cc1cc(CCCC(=O)NCCCN(C(=O)Cc2cc(C)[nH]n2)CCO)on1 C1(COC(=O)NC)CCCCN1C(c1ncncc1Br)=O N1(C(C(C)SCc2ccccc2)=O)CC2CCCC1(CO)C2.c1(C(=O)N)ccsc1 c1(N(C(C2CC(CC)C2)=O)C)cccc(C(c2ccc(Cl)cc2)C)c1 c1(C(N2CC3C(NC(C(C)C(C)(C)C)=O)C3C2)=O)cc2cc(F)ccc2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CCN(C(C(C(C)C)NC(C)=O)=O)C)C(C)C CCC(CC(=O)NC1CC2C(NC(C3CSCN3C(C)=O)=O)C2C1)C1CC1 C12(C(=O)NCCCC3CCCOC3)CC1CN(C(c1cccc(C3CC3)c1)=O)C2 CN1CCC(OCC(N2CCN(Cc3cn(CCCF)nn3)CC2)=O)CC1 N#CC1CCCC(C(N2CC(C3CC3)(C(N3CCN(C4CC4)CC3)=O)C2)=O)C1 C(=O)(CCCCS(C)(=O)=O)N(C)Cc1ccc(CNC(C2=NOC(C)C2)=O)cc1 C1(CC=C)(NC(c2cnc(NC)s2)=O)CCN(C(=O)C(C)(C2CC2)OC)CC1 C=CCC(CNC(=O)CCC(C)C)C(=O)N1CC(C)C(C)(OC)C1 CC(C)C(C(=O)N(C)C)NC(=O)C(O)CNC(C1CC(C)(O)C1)=O NC(=O)CC(N)C(=O)NCC1(c2ccc(F)cc2)CCCC1 CN1C(=O)CCCC1NC(CC1N(C(C2CCOCC2=O)=O)CC1)=O C1(N(C(C(C2CC2)OCC)=O)C)CC2CC1N(C(=O)Cc1ccc(OC)cn1)C2 Cc1cccc(N)c1C(N1CCC(=CCNC(=O)C(c2ccccc2)F)CC1)=O c1(C(=O)NCC2(NC(c3n(CC)ccc3)=O)CCCCC2)ccc2n[nH]cc2c1 CC(C)(C)CC(=O)NC(C(=O)NCC(C)(C)OCC1CC1)C1CCCC1 CC1=NOC(C(=O)NC(Cn2ccnn2)C(=O)N(C)Cc2nnc(O)o2)C1 N1(C(C2(NC(C(C)NC(C)=O)=O)CC2)=O)CCC2(C=CCO2)CC1 c1(CC)ccc(C)c(NC(N2CCOCC2c2noc(C(C)C)n2)=O)c1 Cc1ccc(C(C)C(=O)NC2CC(NC(c3csc(Cl)n3)=O)C2)cc1 C1(S(=O)(=O)c2ccccc2)(C(N2CCc3n(cc(C)n3)CC2)=O)CCOCC1 c1(C(=O)NCCN(C(=O)CC(O)C(C)C)CCC)cccc(F)c1C1CC1 c1(C(N2CCC(NC(C(C)SC)=O)C(O)C2)=O)ncc(P(C)(C)=O)cn1 N1(C(C(CC)NC(C)=O)=O)CC2(NC(c3cc(-c4ccccc4Cl)[nH]n3)=O)CC1C2 N1(C(C)=O)C(=O)CCC1OC(=O)CCC1CCN(CC)C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC(C)C(NC(C2(CN(C)C)CC2)=O)C1 c1(C(=O)NCC(CC)NC(c2cccc(OC)n2)=O)cc(CO)c(C)o1 C(=O)(C(C)(CO)NC(c1ccc(O)nc1)=O)NCC(C)OC c1(C(=O)NCC2CCN(C(=O)Cc3ccc(F)c(F)c3)C2)cnn2c1OCCC2 N1(Cc2ccc(CCOC)cc2)CCN(CC(N2CC(O)C(O)C2)=O)C(=O)C1 Cc1ccc(C(=O)NC2CCCC2NC(C2CCCN2C)=O)c(F)c1F c1(C(=O)NC(C)C(C)NC(=O)CCc2cn[nH]c2)ccc(C(F)(F)F)nc1O CC(C)(C(=O)NCC1(CNC(=O)CCCc2ccccc2)CCC1)C(F)F n1(CC)nc(C)c(CC(=O)NC2CC(F)(CNC(=O)CC3OCCO3)C2)c1C C1(NC(c2cc(CO)on2)=O)CC1C1CCCN(C(=O)Cn2cnnc2O)C1 N1(C(C(c2cn(CC)nc2)(C)C)=O)CC2CCN(C(C34CC(CO)(C3)C4)=O)C2C1 N1(C(C2CN(C)C2)=O)CC(NC(=O)CNS(N)(=O)=O)C(C2CC2)C1 O(N=C1CCCCCC1)CCNC1CC(NC(=O)CC(c2ccc(Cl)cc2)O)C1 c1(C(N2CC(CNC(CC(C)(C)C)=O)C3C2C3)=O)ncn2cc(Cl)ccc12 CC1(C(N2CCC(CO)(CNC(c3ccon3)=O)CC2)=O)CCCS1(=O)=O C1(C(=O)NCc2cc(C(N3CC(OCCCCC)C3)=O)on2)CC2C(C1)C2(F)F c1(NC2C(C)N(C)CCC2)nc(=NCCc2nc[nH]n2)[nH]c2c1CCCCCC2 c1(CC(=O)OCC(CC)=O)cc(F)cc(F)c1 C(=O)(C1CCc2nccn21)N1CCN(C(C(CC)CC)=O)CC1CO Cc1conc1C(=O)N(CCCNC(C1CCC1)=O)CCO S(=O)(=O)(c1c[nH]ccc1=NCC1CCCC(C2CC2)O1)NCC=C(C)C C(C(C(=O)NC1CN(C(C)=O)C(C)(NC(=O)C(C)CC(C)(F)F)C1)C(F)(F)F)OC Cc1[nH]nc(C(=O)NCCOC2CCN(C(c3ccc(Cl)cn3)=O)C2)c1F C1(CNC(C2C(OCC)C2C)=O)Cc2ccccc2CN1C(C1C=CCC1)=O c1(C(=O)NC(c2cn(CCCC(=O)O)nn2)(C)C)cnn2cnnc2c1 C1(NC(c2ncc(OC)s2)=O)CN(C(=O)CCCC(=O)NC2CC2)CCC1(F)F c1(CNC(=O)NCC(C)CN2CCCC2)nc2c(s1)CC(C)CC2 CCC(C)(F)C(=O)NC1CCCC1NC(c1cn(C2CCCC2)nn1)=O C1(C(=O)NC(COC(C)C)C(C)C)CCC(NC(C(COCC)N(C)C)=O)CC1 N1(C(c2cn(CC(C)C)nc2)=O)CC(CNC(=O)CCC#N)CC1C N1(C(C(CC=C)NC(=O)OC(C)(C)C)=O)CC2CCCC(NC(=O)C3CC3)(C2)C1 C(=O)(C1CCCc2n[nH]cc21)N1CCCCC(NC(c2c(C)nc(Br)o2)=O)C1 N1(C(C(C)OCC=C)=O)CC2(C(CO)C2)CC1(C)CNC(=O)CSC(C)C.C1(O)CC1 c1(OCC)nc(N2CCN(C(=O)NCc3cccc(I)c3F)CC2)ncc1Cl c1(C(N2CC(CC(CNC(C(CC=C)CC)=O)(C)C)C2)=O)c(Cl)oc2ccccc12 O(C1CCOc2c(Br)cccc21)CC12C(C)(C)C(CC1)CC2 CC1NC(=O)CCC1CN(C(C)C(=O)O)C(c1ccccc1)=O c1(NNC(C2(c3cn(CSCCCc4onc(C)n4)nn3)CC2)=O)cnn(C)c1C.S.C N1(CC(=O)NCC2CCN(C(C3(C(C)C)CC3)=O)C2)CCN(C)CC1 N1(C(c2cn(C)nc2Cl)=O)CC2CC(NC(C3(F)CCCCC3)=O)CC2C1 C1(C(N2CCC=C(C(=O)Nc3cncs3)C2)=O)CCC2CCC(=O)N2C1 c1(SC)cc(C)c(C(N2CCC(C3CCCCN3C(=O)CC=C(C)C)C2)=O)o1 c1(C(=O)NCCCC2N(C(C3(F)C(C)OCC3)=O)CCC2)ccc2cccnn12 c1(C(N2CC(O)(C(C)NC(C(C=CC)O)=O)C2)=O)cn(C)cc1C c1(C(=O)NC2CN(C(c3cc(CC(C)C)on3)=O)C(C)C2)ccc(Cl)c(Cl)c1O N1(C(CC(CN(C)C)O)=O)CC2CCC(C1)N2C(=O)CCC1CCCC(=O)N1 O=C(C1SCCc2ccccc21)NC1CC(F)(CNC(C2(F)CC2)=O)C1 C(=O)(CCN=c1[nH]ccs1)NC1CCC(CNC(C(c2cccnc2)OC)=O)C1 C1(CC)CCC(C(N2CC(NC(c3nncs3)=O)C2)=O)O1 C12(OC)CCC(C(N3CCOCC(CNC(=O)C(C)C(C)(F)F)C3)=O)(CC1)C2 C1(NC(COCCCC)=O)CCCC(NC(c2ccc(C)cc2F)=O)CC1 C(=O)(C1=CNC2=NCCCN12)NC1C(CNC(c2onc(C)c2C)=O)C1 Cc1c(C#N)c(NCCNC(=O)C2=C(Cl)CC2)nc2ccccc12 C1(NC(c2cc(C)on2)=O)CCN(C(c2cn(C)nc2C(F)(F)F)=O)CC1CO N1(C(c2cc(C)ncc2)=O)C2CCC1C(NC(C1CCC1(C)C)=O)C2 C1(CC(=O)NC2CCN(C(C(C)(C)C)=O)CC2O)CCCC(C)(C)CC1 Cc1cccc(C(N2CC(O)CC2CNC(=O)CCOc2ccccc2F)=O)n1 c1(C(N2C(C(=O)Nc3cc(CO)ccn3)C=CC2)=O)c(Cl)cccc1Br C1(NC(C(CC=C)OC)=O)(CNC(=O)C=CC)CCCCC1C c1(C(=O)NCC(C(C)OCc2ccccc2)O)coc(S(=O)(=O)N(C)C)c1 Cc1onc(C2CC2)c1C(=O)NCC.N12CCC(CC1)C2.C1(=O)CC2(CC2)N1C C=C(C)CCCC(=O)N1CCC(NC(=O)C(c2cnn(C)c2)OC)C(C)C1 Fc1cnccc1N1CCCC(NCc2coc(-c3ccccc3)n2)C1 C(CCCC(=O)NC(c1ccc(-c2nc(C)c(C)[nH]2)s1)C)SC c1(NCCC(=O)N(C2CCN(C(c3ccc(Cl)[nH]3)=O)C2)CC)ccccn1 Cc1ccc2c(C(N3CC4CCC3C(NC(C3CCO3)=O)C4)=O)c[nH]c2c1 CC1(CCNC(=O)CCCN(C2CC2)C2CC2)CCN(C(=O)CCn2ccnn2)C1 c1(C(=O)NCC2(F)CN(C(C3C(C)CCO3)=O)C2)cc2ncccc2o1 C12(NC(C(CC)OCC)=O)CCCC1CN(C(c1ncc3ccccn13)=O)C2 c1(C(=O)NC(C2CCN(C(c3n[nH]c(C)c3Br)=O)C2)C)cc(F)ccc1N N1(C(C)=O)CCc2ncccc2C1C.O(C=CC(=O)NNC=O)C(C)C N1(C(C(C)NC(C)=O)=O)CCC2(CC2NC(c2cccc(C)c2)=O)C1 C1(C(N2CCOCC(CC)C2)=O)CC2(CCN1C(=O)Cc1ccsc1)CC2 c1(NC(C2CC2C(=O)Nc2nccnc2Cl)=O)ccnc(Cl)c1 C1(C)(C(N(C2CCSC2)CC(N2CCN(C(C)C)CC2)=O)=O)CC2C=CC1C2 c1(CC(N2CCC(CN(C)C(c3cccc[n+]3[O-])=O)C2)=O)cc(O)nnc1O Cc1cc(C(N2CCOC(CC3CCCOC3)C2)=O)c2ccc(C)c(C)c2n1 c1(C(c2nnnn2Cc2nnn(C)n2)NCC=CCSC)ncccc1Cl N1(C(c2ccn(C)n2)=O)CCCC2CN(C(=O)CCc3cc[nH]n3)CCCC12 N(C(=NCCF)N1CCC(CC(C)(C)C)C1)CC(=C)C c1(C(=O)NC2(CNC(C(C=C=C)C)=O)CCOCC2)ccc2c(c1)CN(C)C2 N1(C(c2n(C(C)C)ncc2)=O)CC(F)(F)CC1CNC(=O)CN1CCN(C)CC1 c1(NC(C(Cc2ccoc2)NC(c2c(CC)[nH]cc2)=O)=O)cc(C)c(C)cc1C c1(OCC)nc(C(=O)N(CCCNC(=O)C(C)(F)c2ccccc2)C2CC2)ns1 C(CCNC(=O)CCc1cnoc1)(C(C)C)NC(CCOCCC)=O Cc1ncc2n1CCC(NCCCC1CCOC1)C2 c1(CC(N2CCC(NC(C=CC(CC)C)=O)C2)=O)c[nH]c2c(C)cccc12 c1(C(=O)NC2CCN(CC)C2)cc[nH]c1C(=O)CC.C(C(C)N(CC)CC)N CCCCC(C)CCC(=O)NCC(C1CCCC1)NC(=O)C(C)(C)C1CCCCC1 Cc1nc2cc(CC(N3C4CN(C(c5c[nH]c6cccnc56)=O)CC34)=O)ccc2o1 Cc1cc(C)c(C(=O)NC(Cc2cn(C3CCCN(C)C3)nn2)C(=O)O)s1 C1(NC(C(=O)NC(COCC)C)=O)CC(C)CCC1C(C)C c1(C(N(c2ccccc2Br)C(C)C)=O)cc2c([nH]1)CCCC2=O c1(CC(=O)N(CCN(C(C2C(OC)CCC2)=O)C(C)C)C)nn(C)cc1Br Cc1ccc2c(c1)SC(C(N1CC3CC(Nc4cc(C(C)C)ncn4)C3C1)=O)C2 Cc1ncc(CN(C)C(C2CCC(C#N)C2)=O)c(O)n1 CCC(O)C(C)(C)C(=O)NCC(CC1CC1)C(=O)NCc1ccco1 Cc1oc(CNC(=O)C=C2CCC2)nc1C(=O)NC1(CN2CCC2)CC1 c1(C(=O)OCc2c(SC(C)C)nc3sccn32)cccc(C#CCO)c1 Cc1cccnc1C(=O)NCCCC(C)NC(=O)CNC(=O)CC1CCCC1 Cc1cccc2nc(N3CC=CC(NC(c4cc[nH]c5nccc4-5)=O)C3)oc12 N1(C(C(C)OC)=O)CCCC2(CCCN(C(=O)C(c3ccc(F)cc3)C)C2)C1 CC(C)C(C)(CNC(=O)C=CCN(C)C)NC(c1cnn(-c2ccccc2)c1)=O C1(OC)CC(C(N2CC(n3cc(CN4CC5CC5C4)nn3)C2)=O)C12CCC2 C1(C(C)C)CCC(CC(=O)N(CC(C)N(C(=O)Cc2nocc2C)C)C)CC1 c1(C(N2CC(NC(C3CC4C=CC3C4)=O)CC(OC)C2)=O)cc2ncccc2[nH]1 C(c1cnccn1)=CC(=O)NC(CCSC)C.C1(=O)CCCN(C)CCN1 c1(CC)ccc(O)c(C(=O)NCC(CO)NC(c2cncc(C(F)(F)F)n2)=O)c1 C1(C(NNC(c2c[nH]c(=NC)s2)=O)=O)CCc2cc(Br)ccc2C1 c1(N2CC(C)(C)C(O)CC2)nc(=NCc2cnc[nH]2)[nH]c2cc(Br)ccc12 c1(C(=O)NC2CC(C(C(=O)NC3(CC#C)CC3)F)C2)ccc(CF)cc1 c1(C(=O)NCC(C)N(C(C(CC)C)=O)C)cc(C)nc2c(C)c(C)nn12 C1(C(=O)NC(CC=C)CNC(=O)C=CSC)OCCOC12CCC2 c1(CCCCC)ccc(C(=O)N(C)CCOCCN(C(=O)CCSC2CC2)C)o1 C12(NC(c3c(C)ncnc3C)=O)CCCC1CN(C(=O)CC1CCSCC1)C2 N1(C(C(=O)NCc2cccc(NC(C)(C)C)c2)=O)CCc2ccc(F)cc21 N1(C(C2(NC(c3cc(C)ns3)=O)CCOCC2)=O)CCCSCC1C C12(NC(=O)CS)COC(C1)C2.c1(C(C)O)ncc(C(=O)NC2CCOCC2)s1 C1(C(=O)NC2C(NC(C3CCC(=O)N3)=O)C2)CCC2(CC1F)OCCO2 C12(NC(c3n(CC#N)ncc3)=O)CCN(C(=O)CCn3cncn3)CC1C2 c1(C(CC)C(=O)NCC(C)CNC(=O)C(C)=C2CC2)ccc(Br)cc1 S(=O)(=O)(c1ccc(C#N)c(N2CCOC(C)CC2)c1)N1CC(C#C)OCC1 CC1(CNC(c2c(Cl)nsc2Cl)=O)CCCN(C(c2cnn[nH]2)=O)C1 c1(C(=O)NC2C(CNC(=O)C=CCF)CCC2)ccccc1-c1nc[nH]n1 C=CC1(O)CCN(C(c2ccc(OCC)c(Br)c2)C(=O)NCCC2CC2)C1 c1(C(=O)NCC2CCC(NC(Cc3c(C)non3)=O)C2)cnc(N)c(Cl)c1 c1(C(N2CC(C=C)(C(=O)O)C2)=O)nn(C)c(Cl)c1CC CC(C)CC(C(=O)N1CCCC(N(C)C)CC1)ONC(=O)CCc1nccs1 CC1(C)CCCC(C)(NC(=O)CCC2CCCN2C(=O)C=CCF)C1 C1(CC(=O)N(CC(C)OC)CC)CC2(C1)CN(C(=O)CC1C(=O)NN=C1C)C2 C1(CNC(C2(O)CCC2)=O)CCCC2(CN(C(=O)CSCc3ccccn3)C2)O1 C1(C)CN(C(=O)C(C)CC)CC(C)(C)C1.N1(CCC)CCC(CNC(=O)CC)CC1 C1(C(N(C)CCOCCNC(=O)CNc2nccs2)=O)C=CCCC1 c1(C(=O)NCCC2C(C)CN(C(C3CN(C(N)=O)C3)=O)C2)nn(C)cc1[N+](=O)[O-] Cc1ccccc1C=CC(N1CC(CO)CC1C1(NC(=O)CC2CCC2)CC1)=O C1(NC(C(C)Cc2cnn(C)c2)=O)CC(F)CN(C(C2(CC3CCC3)CC2)=O)C1 c1(CS(N2CC(COC)OCCC2)(=O)=O)nc2cc(F)ccc2s1 c1(C(=O)NC2CC3(CN(C(c4cn(C)nc4)=O)C3)C2)cc(O)c(F)cc1N c1(OC)ccc2ncccc2c1C(N1CCC(NC(c2cc(N)ccn2)=O)C1)=O c1(C(=O)NC2C(C(=O)NCC3CCN(CC)C3)OCC2)cncc(OC)n1.OCC C1(OC2CN(C(C3C(CC)CC3)=O)C2)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1 C1(C(=O)NCCCOCCC(F)(F)F)CCOC2(CCOCC2)C1 N1(C(c2c(C)cc(I)cc2)=O)CC2(C1)CN(c1ncnc3cnn(C)c13)CCO2 N1(CC)CCCC1CNC1(CC(=O)NCCc2cnn(C)c2)CCOC1 N1(C(C2C=C(C)CS2)=O)CC(O)CCC1C(=O)NCCn1cncn1 N1(CC(Cc2ccc(F)cc2)N(C2CC(C)(C)C2)C)CCCC(COC)C1 C(CCN=c1[nH]c(=NC2CC(NC(N)=O)C2)[nH]c2c1CCC2)OC1CCN(C)C1 C1(NC(C=NOC)=O)(COC)CCN(C(C23CC(C2)C3)=O)C1 N1(C(CCC#C)=O)CCC(C(=O)NC(C)CCC2CC2)CC1C CC1=C(C)CC(C(=O)NCC(C)(Cn2cccn2)NC(=O)CC(C)C(C)C)CC1 Cc1cc(C(=O)NC(C2CC2C(=O)NCC(C)F)C)n[nH]1 CC1(C(=O)NCCCN(C(c2cnn[nH]2)=O)Cc2ccccc2)CCCOC1 N1(C(C2(OC(C)=O)CC2)=O)CCC2CCN(C(=O)C=C(C)C3CC3)CC2C1 c1(C(C(=O)NCCN(C(=O)CCCc2cscn2)C)=O)ccc(F)cc1 C(=O)(CCCC(=O)NCC(F)CNC(=O)CC1C(=O)N(C)N=C1C)NCC CCC(CC(F)(F)F)C(=O)N1CC(NC(C2CN(C(N)=O)C2)=O)C2(CCC2)C1 C(=O)(C(=O)N=S(C)(C)=O)NCc1c(OCCOC)cccc1 N1(C(C=C(C)C(F)F)=O)CC2(CCN(C(=O)CCn3cccc3)CC2)CC1C c1(C(=O)NCC(CC)(CC)NC(=O)CCN(C)CCO)ccc(Br)cc1Cl C1(CNC(CC=CC=C)=O)CN(C(=O)C=Cc2ccc(SC)s2)CC1(C)C C(C(CC(C)C)C(=O)NCCn1ccc(C(N2CCC(O)C(CO)C2)=O)c1)OC N1(C(CNC(CC)=O)=O)CC(NC(=O)C=Cc2cncnc2O)CC(C)C1 c1(C(N(C)CC2CCCCN2C(c2sccc2CC#N)=O)=O)ccccc1C#N N1(C(CN(C(C(C)C)=O)C)=O)CCC(C)(CCNC(C2CCN2S(C)(=O)=O)=O)C1 C(C(N=[N+]=[N-])C(=O)NC1(CNC(C2CCN2C)=O)CCCCC1)OCC C=CCC(C)(C)CC(=O)N(C1CN(C(=O)CCCn2cncn2)CCC1O)C c1(Cc2c(C(=O)NC3CC3CF)nccc2)nc(-c2ccccc2)ncc1C Cc1cc(C(N2CCN(c3ccc(F)cc3)C(C)C2)C(=O)NC(C)C)cc(F)c1 Cc1cc(O)ccc1-c1ccc(C(N2CC(O)C(F)C2)=O)c(C)n1 c1(CSC)cc(O)nc(-c2cccc(C(=O)Nc3cncnc3)c2)n1 N1(C(=O)NCC2(c3coc(O)n3)CC2)CCCC(O)(C2CC2)C1 CC1=C(C(=O)N2CC(C(F)Cc3cn(-c4ccccc4CO)nn3)C2)COCC1 C1(NC(C(C(=O)OC)OC)=O)CC(C(N2CC(O)CC(O)C2)=O)C12CCC2 N1(C(C2C(C)OCC2)=O)CCC(C)(CNC(=O)CC=Cc2ccccc2)CC1 Cc1ccc(CCOCSc2ccccc2C)cc1.N1(C)CC1 N#Cc1ccccc1C=CC(N1CC2(CC(CNC(C3CC3F)=O)C2)C1)=O C1(CNC(c2cccc(OC(F)F)c2)=O)CN(C(=O)CSc2nncs2)C2CC12 CC1COc2ccc(C(N3CCC(NC(C4C=CC=CC=C4)=O)C3(C)C)=O)cc21 c1(C(=O)OC)cccc(OC2CN(Cc3cnsn3)C2)c1 C(=O)(C(C)C(O)C(C)CC)N1CC(C(N)=O)(CNC(C(C=C)(C)CC)=O)C1 N1(C(c2[nH]c(=NCC)sc2)=O)CC(C)CN(C(c2cc(O)nc(O)n2)=O)CC1C C1(NC(C(C)=C2CC2)=O)CCC2(CC1)CN(C(=O)C(F)CCC(C)(C)C)C2 c1(C(N2CCC3CN(C(C(C)SCCCC)=O)CC32)=O)cc2nc[nH]c2cc1N CC1CC(CC(=O)NCC2(CCNC(c3cc[n+]([O-])cc3)=O)CC2)CC(C)(C)C1 c1(C(=O)NCC(C)CNC(C2CCCC2F)=O)cc(Cl)c(Br)cc1F N1(C(c2ncn3c2CCC3)=O)CC2CC(NC(=O)C(F)(F)C(F)F)CC1C2 n1(NCCC(=O)N(S(C)(=O)=O)CCOC)cc(CC2(O)CCSC2)nn1 C12(NC3CCCN(C(=O)OC(C)(C)C)C3)COCCC1CN(C(C1CCC1)=O)C2 c1(OC)ccccc1C(=O)NCC1(C(=O)NC2(CSC)CC2)CC1 C1(NC(c2c(C)n(C(C)C)cc2)=O)C2CC1N(C(=O)C(c1ccccc1)F)C2C C(=O)(CCS(N)(=O)=O)N(C1CCN(CC(c2ccccc2)O)C1)CCC C1(C(C)C(=O)NCc2ccoc2)CCN(C(c2cnn[nH]2)=O)C1 C(=O)(C(C)(C)C(=O)N1CC2C(CNC(c3cnc(O)c(F)c3)=O)C2C1)NC C12(NC(c3ccnc(C)c3C)=O)CCOCC1CN(C(=O)Cc1cnns1)C2 C1(C(N2CC(NC(C3CCCO3)=O)C(n3ccnn3)C2)=O)Cc2nncn2C1 N1(C(C(=O)NCC)=O)CCC(n2cc(CNC(=O)C(C)OCC(C)C)nn2)CC1 C12(C(=O)NC3CCCC(NC(CCCC=C)=O)C3)C3C4C1C1C2C3C41C c1(C(=O)NCC2CN(C)C(=O)C2)cccc(CNC(=O)Cc2ccc(O)cn2)n1 c1(C(N2CCN(C(C(C)O)=O)C(CC(F)F)C2)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(c2ccc(C)cc2)=O)CCCCC12CN(C(C1CCCN1S(C)(=O)=O)=O)C2 C1(F)(C(N2CC(C)(CC=C)C2)=O)CCCN(C(C2CCC(N=[N+]=[N-])C2)=O)C1 C(=O)(NNC(=O)c1cn(C)nc1-c1ccc(C)o1)NC(C(OC)OC)C C(Cc1ccccc1)(CCNC(C1CC(N(C)C)C1)=O)NC(COCC)=O C1(C(=O)NCC(CC)CC)CC12CCN(C(C1CC(C)(C)CO1)=O)CC2 N1(CCNC(c2cc3ccc(Cl)c(F)c3o2)=O)CCCC2(CC=CCO2)C1 N1(C(C(C)(C)SC2CCCC2)=O)CC2CC(NC(C3CC4(C3)CC43CC3)=O)C1C2 c1(C(N(C2CCN(C(CCN(CCCCC)C)=O)C2)CC)=O)ccc(O)c(N)n1 CC1CC(C)N(C(c2cn(C)c(O)n2)=O)CCN1C(=O)CC[SH](c1ccncc1)CCO C1(NC(c2n(C(C)C)ccc2)=O)CN(C(=O)CCC(C)(C)C)CCC1(C)C C(CNC(=O)C(F)(F)CC1CC1)(CC(C)C)NC(C1C(c2nnc(C)s2)C1)=O C(=O)(C1=C(C)CCC1)NC1(C(N(CC#C)CC2CCCO2)=O)CCCC1C c1(C(N(CCOCCC(=O)N(c2cccc(O)c2)CC)C)=O)ncc(F)cc1C C1(NC(C(C)=C(CC)C)=O)CCN(C(C2CCN(c3ccncc3)C2)=O)C(C)C1 n1(CC)nnnc1C(CCC1CC1)NCc1ccc(-c2ccccc2)s1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCC(F)(F)F)N1CC(CC(=O)OC)C1 C1(C(CC)C)CCN(c2cc(N3CCC(C)(c4cccc(C)c4)C3)ncn2)CC1 N1(C(c2ccn(CC)c2C)=O)CCCC2(C1)CN(C(C1CC1C)=O)CCO2 O(N1CCC(NC(=O)CCCC(C)NC(C2CCC(C)(O)CC2)=O)CC1)CC c1(C(=O)NC(c2cn(C(c3cc(F)cc(F)c3)C)nn2)C)ccc([N+](=O)[O-])[nH]1 CC1C2CCCN1Cc1ccc(o1)C(=O)N2.C1(C(N(C)C)=O)CC(F)C1 C1(C(N(CCN(C)C(C2CC3(CCCO3)C2)=O)C)=O)CC(=O)CC12CCC2 c1(C(=O)NCC2CC(NC(=O)CCSCC(F)(F)F)C2)cn2ccccc2n1 c1(C2CCCN(C(c3ccc(-c4ccncc4)cc3)=O)C2)cccc2cc[nH]c12 c1(C(N2CC(C(=O)NC3(C#C)CCOC3)C(OC)C2)=O)cccc(C#N)c1C C(=O)(C1=CCOCC1)NCC1C(NC(C2CN2C)=O)CC1.C(C)(C)(C)OC(=O)N.CO C1(NC(C2N(C)C(=O)NC2)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CC12CC2 N1(C(=O)CCSC(F)(F)F)CCCCC1C1CCCN1C(C1OCCO1)=O c1(C(=O)NCCOCCNC(C2C(C)(CC)C2)=O)cn(CC(N)=O)nn1 C1(CCC)CN(C(c2cnn(C)c2SC)=O)CCN1C(c1cc(C)c[nH]1)=O N#CC1(C(=O)NC2CC(NC(=O)CCn3cnccc3=O)C2)CC=CC1 Cc1cccc(Br)c1C(C(=O)NCc1cnc[nH]1)NC(=O)CC1CCCC(=O)N1 c1(C(=O)NC2CC(C(C(=O)N(C(C)C(C)C)CC)F)C2)cccc(O)n1 N1(C(C2CCN(C(c3cn(C)nn3)=O)CC2)=O)CC(O)CC(C)(C)C1 C(C)(C)(CCNC(c1ccc(OCCC)s1)=O)NC(C(C)OCCCC)=O.C(C)=O C(C(CNC(=O)CC1CCCCCC1)C(F)(F)F)NC(C(C1CC1)SC)=O S(=O)(=O)(c1cc(F)ccc1F)NC1C2CN(c3nccc(SC)n3)CC21 C(=O)(C1=CSCCO1)N(CCCCN(C(=O)CN1CCCCCC1)C)C c1(C(=O)NC2C(C(=O)NC(c3ccccc3)(C)C)C2)cncc(F)c1 C(=O)(C1CC(=O)Nc2ccccc21)NCC1C(OC)CCC1 CC1C(C(=O)NCCCS(N)(=O)=O)CCN1C(C1CCN(C)CC1)=O C(=O)(C1=NOC2COCC12)N1C(c2cn(C3CCCC(C)C3)nn2)CCC1 N1(C(Cc2ccn(CC)n2)=O)CCCN(C(C23CC2COC3(C)C)=O)C1CO C1(NC(c2cnsc2)=O)COC2(CCN(C(=O)C(F)(F)CO)C2)C1 C1(N(CCCn2c(N)ccn2)C(C2CCOCC2)=O)CCN(c2cccnn2)CC1 C(=O)(C#CC1(C)CCCO1)NC(CCCNC(C(C)=C1CC1)=O)C c1(C(=O)NCC(C)N(C(c2cc(Br)n(C)c2)=O)CC)cccc2c1OCC2 C(=O)(CC(C(C)CC)NC(=O)CCC(=O)N(C)C)NCC(CCC)(C)C CCC(CC)(CC)N=c1cccc(S(=O)(=O)NCC2CCCC3CC23)[nH]1 CON=CC(=O)N(CCC(C)NC(c1cnc(COC)s1)=O)C N1(C(C(CC)C)=O)CCC(c2n[nH]c(CNC(=O)COC3COC3)n2)CC1 CC1(C)CN(C(=O)C2=CCCCC2)CCC1NC(=O)CCNc1ccccn1 CC(O)C(O)C(=O)NCCCNC(=O)NCCCc1ccccc1F C1(NC(c2ccc(Cl)cn2)=O)CCN(C(=O)CC2CCC(C(F)(F)F)O2)CC1 C(CO)(C(F)(F)F)NC(C1CC(C)N1C(=O)CN1CCCCC1=O)=O C12(NC(C(C)n3ccnc3)=O)CC(CNC(=O)CCn3ccnc3)(C1)OC2(C)C C1(CNC(c2c(CC)n(C)nn2)=O)C(O)C(O)CN1C(=O)CC1CCCC1OC C1(NC(c2ncn(C)n2)=O)C2CCN(C(c3c[nH]c(=N)nc3C(F)F)=O)CCC12 c12ccc(cc1)[nH]2.C1(C(C)NC(=O)OC(CC)CSCCC)CCC(=O)N1C c1(C(=O)NCC2CCCN2C(=O)C(F)=CCCF)ccc(F)c2cccnc12 c1(Oc2ccc(C(N3CCC(NC(=O)OC)C3)=O)cc2)ccc(F)cc1C N1(C(N(CC(CC)(O)CC)C)=O)CCC2(C1)OC(=O)NC2C.C(C)(=O)OC C1(NC(c2nc(C)sc2)=O)CCOC(C(=O)NCCc2ccco2)C1 c1(OC)ccc(C(=O)N(CCCNC(C2C(C)C2C)=O)C2CC2)c(F)c1N CC(CNC(=O)Cc1cnns1)C(=O)NC1(C2CC2)CC1 C12(C(N(CC(CC)CC)CCC)=O)C3C4C5C3C1C5C24.C1CCNC1=O O=C(CCC(=O)c1ccccc1Br)NC1(CNC(C2CC2F)=O)CCC1 C(C)(CNC(=O)CN1CC2CC2C1)(CNC(=O)C(C)c1ccco1)OC c1(C(=O)NC(C2CCCCC2)C(C)NC(CC)=O)cc(C)cc(OC)c1C N1(C(CN2C(=O)CCCC2)=O)CC2CCC(C1CO)N2C(c1cc(Cl)cnc1O)=O c1(C(=O)NC(C(=O)OC)Cn2cncn2)c[nH]c2cc(F)ccc12 CCC(CC)CC(F)C(=O)NC1CN(C(=O)Cc2ccccc2)CC1C(F)F C(CC)(C(=O)N(CC(=O)N(CCCOCC#C)C)C1CCC1)=CC N1(Cc2ccc(OC)cc2)CCCC(NC(=O)C(C)Oc2cccc(C)c2)C1C C1(CC(=O)NC2CC(n3cnnc3)C2)COCCN1C(c1ccc(OCCO)s1)=O c1(OCCC)nc(C)ccc1NC(=O)NNC(=O)c1cccnc1O N1(C(Cc2ccc(C)s2)=O)CCN(C)C(C(=O)N(C)Cc2nc(C)ns2)C1 N1(C(c2c(C)ncnc2C)=O)CCC2(CCC2NC(=O)CCSCC(N)=O)CC1 c1(C(N2CC(CNC(=O)COCCF)C3C2C3)=O)cccc2c1OCCN2 c1(CCC(=O)NC2CC(NC(C3(C)CC3(Cl)Cl)=O)C2)cnc2n1CCOC2 Cc1ccc2c(c1)C(NCc1cccc(Br)c1I)C(C)C2 c1(C(N2CCCCC2CC(C)C)C(=O)NCCC)ccnc(OC)c1F N1(c2nccc(CC(=O)OC)n2)CC2CC(NC(=O)C(C)SC)C2C1 c12ccc(cc1C)[nH]c2=O.C1(C(N(CCCC)CC)=O)CSCN1C(C)=O N1(C(c2c(C(C)(C)C)c[nH]c2)=O)CC(NC(=O)CCc2nc(=N)[nH][nH]2)CC(O)C1 C12(C(N(C)CC=CC(=O)NOCC3CCOC(C)(C)C3)=O)CCC(O)(CC1)CC2 CCCCC(=O)NCC1CCC1CNC(=O)C(C)Sc1nnnn1C1CC1 n1(CC)cc(CC(=O)NCCC(C)N(C)C(C2CCC(=O)N2)=O)cn1 C=CCC(C(=O)NCCCN(C)C(C12CCOC(C)(C1)C2)=O)C(C)C C#CC1CN(C(=O)C(C)n2cccc2)CCN1C(=O)CC(C)SC C1(C(=O)NCc2ncc(C(=O)NCC3(OC)CCC3)cn2)CCOC(=O)CC1 CC12CC3CC(C(=O)NC4CC(NC(C5(CCO)CC5)=O)C4)(C1)CC(C)(C3)C2 c1(C(=O)O)ccc(S(=O)(=O)N2CCOCC(O)C2)c(Cl)c1 N1(C(CCSC)=O)CCN(C(=O)COCC(C)C)CC(C)(F)C1 C1(CNC(CC(CCC)C)=O)CCC2(CN(C(=O)C3=C(C)CC3)C2)O1 C(=O)(CC1CCc2ccccc21)NC1CC(CNC(CCS(=O)(=O)N(C)C)=O)C1 C1(C)(NC(C(C)N(C(C2CN(CC)C(=O)C2)=O)C2CC2)=O)CCCC(C)(C)C1 N1(C(C(N2C(CC)CCC2)=O)=O)CCN(C(c2cnc(N)c(N)c2)=O)C(CF)C1 N1(C(C2CC(=C)C2)=O)CC2(CC(NC(c3snnc3OCC)=O)C2)C1 C12(C(=O)NC3CN(C)C3)CC(n3cc(CNC4CCCC4)nn3)C1C2 c1(C(N2CCC(CNC(C34CCCC(CO3)C4)=O)C2)=O)ccc2c(n1)NCCO2 C1(NC(c2cncc(N(C)C)c2)=O)CCN(C(c2ccc(CO)s2)=O)CC1F C1(CNC(C2C(Cl)(C(=O)OCC)C2)=O)(NC(c2ccccn2)=O)CCCCC1 N1(C(c2cc(-c3ccccc3)cn2C)C(=O)NC(C)C)CCS(=O)(=O)CCC1C CC1CCc2[nH]c(C(=O)NCCC(C)(C)S(C)(=O)=O)cc2C1 c1(C(N2C(CC)C(NC(C3CC3C)=O)CC2)=O)cc(Br)c(C)nc1OC C1(NC(Cc2ccn(CC)n2)=O)C2CN(C(C)C)CC12.C1(CO)C(C)N1 C1(c2ccccc2)(NC(C=C(C)C(C)C)=O)CCN(C(C2CC2(F)F)=O)CC1 C1(NC(CCC=C)=O)CC(C)N(C(c2ccc(-c3noc(CC)n3)cc2)=O)C1 Cc1cc(C(N2CCN(C(c3sc(F)cc3Cl)=O)C(C3CC3)C2)=O)cn(C)c1=O C(C(=O)N(CC(=O)N(C(COC)CC)C)CC)(C1CCC1)OCC N1(C(c2n(C)nnc2)=O)CC(F)(F)CC1CCNC(c1c[nH]nc1[N+](=O)[O-])=O N1CCc2ccccc2C(NC(C23CC2C3)=O)C1.Cn1c(O)nc(N)cc1=O C(CC(C)C)(C(=O)NCCc1cnco1)NC(C(C1CCC1)OCC)=O C1(NC(c2ccc(C(C)(C)C)[nH]2)=O)CN(Cc2ccc(CBr)cc2)CC1F C1(C(=O)NCC(C(=O)OCC)C)CCN(C(C2CC2CC(C)C)=O)CC1 C(=O)(C1=CC(C)(C)C1)NCCCCCCNC(C(N(C)C)C1CC1)=O N1(C(c2cc(OC)no2)=O)CC2CCC1C2NC(=O)CCC(C)SC c1(C(=O)NC2CC(F)(CNC(C(C)NC(C)=O)=O)C2)ccc2nn[nH]c2c1 CCCCC(CC)CC(=O)NCCCCCNC(=O)CCn1ccnc1C c1(C(=O)NC(CNC(C2CCCC3(CC3)C2)=O)C2CC2)cc2ncccc2o1 c1(C(=O)NC(CNC(C(C)NC(CC)=O)=O)CC)ccc(C#N)nc1C Cc1nc(C(=O)NC2CCC2NC(C2CC(=O)N(C(C)C)C2)=O)ccc1Br C(C(=O)N=c1cc(C2CC2)[nH][nH]1)c1cccc(OC)c1F Cc1cc(C(=O)N(C(C)C(=O)Nc2ccc(Cl)nc2)C2CC2)ncn1 C1(C2CCN(C(c3cscc3Cl)=O)CC2)(NC(C2CCC2F)=O)CC1 Cc1oc(Br)cc1C(N1CCCC(CNC(C2(N=[N+]=[N-])CC2)=O)C1)=O C1(C(=O)NC(C(C)NC(c2[nH]c(=NCC)sc2)=O)(C)C)CCc2c(nnn2C)C1 N1(C(C2(C=C)CCN(C(c3ncccc3Cl)=O)C2)=O)CC(C)(C)OCC1C c1(C(=O)NCC2C(NC(c3c(CC)noc3)=O)CCC2)cc(OC)cc(CC)c1 C1(C)(CCC)C(=O)NCCN1C(C1COCCN1C(c1c[nH]nc1C(F)F)=O)=O N1(C(C2C(CC)C2)=O)CCN(C)C(CNC(=O)COC(F)(F)F)C1 c1(C(C)=O)ccc(NC(c2cncc(NC(C3CC4CC4C3)=O)c2)=O)c(Cl)c1 CC1(C2CCN(C(=O)CC3C4CN(C(=O)C(F)OC(F)(F)F)CC34)C2)CC1 c1(C(N2CC(C(N(CC(CC)C)C)=O)OC(C)C2)=O)ncc(C#N)cc1C c1(CC)cccc(C(=O)NC(C)(CNC(C2CC(C(C)C)=NO2)=O)CC)c1N c1(OC)ccc(C(C)C(=O)NCC2CCN(C(=O)C3=C(Cl)CC3)C(C)C2)c(C)c1 N1(Cc2cnn3c2CN(c2c(C)cncn2)CC3)CCc2nc(C)nc(O)c2C1 C12(NC(C(C)C3CCOC3)=O)CC(C(=O)NCC3CCC(O)C3)(C1)C2 c12ccc(s1)[nH]c2=O.c1(C2CN(C)N2C)ccsc1.C(C)(C)(C)OC=O.C(C)(=O)N C1(CCO)(NC(CN(CC)CC)=O)CN(C(=O)CC(C)C2CCCO2)C1 Cc1cccc(C2(NC(=O)C(=O)Nc3cncc(N)c3)CCC2)n1 C(C(CC(C)C)C(=O)N1Cc2cccnc2C1)NC(c1ccc(C)nn1)=O c1(C(N2CCCC2C2CC2(F)F)C(=O)NC(C(=O)OC)C)cc(C)cs1 N1(C(C(C)C)=O)CC2(CC(NC(C3(CC4CC4)CCCO3)=O)c3nccn32)C1 C1(CC)CN(C(C2C(C)(C)C2(C)C)=O)CCC1NC(c1ccc(Br)cc1)=O CC1CC(NC(c2ccc(CO)c(F)c2)=O)CN(C(c2cc(F)ccc2Cl)=O)C1 C1(NC(=O)CCCCCF)CC1C1CCN(C(=O)CC2CCC(F)(F)CC2)CC1 N1(C(CS(=O)(=O)NC)=O)CCN(C(c2ccc(C(C)=O)[nH]2)=O)C(c2ncc[nH]2)C1 C1(CCNC(CC(=O)NCC)=O)CN(C(=O)C(c2cccc(Cl)c2)C)CC1C C1(NC(=O)Cn2cc(Cl)cn2)CN(C(c2cc3c[nH]cnc-3n2)=O)C2(CCC2)C1 CCC(C(=O)NC(C)(CNC(C1CCN(C)C1)=O)C1CC1)n1cccn1 C1(CCNC(C2(C)CCN(C)C2)=O)CCCN(C(=O)CCc2ccn(C)c2)CC1 Cc1cc(CNC2CCCN(C(c3cc(C(N)=O)ccn3)=O)C2)c(C)[nH]1 C1(C(=O)OC)CC2(CCC(NC(=O)NCCn3ccnc3C)CC2)C1 C1(CNC(c2c(C)cn(C)n2)=O)CC(NC(=O)Cc2cncs2)C12CCC2 CC#CCC(C(=O)NC(CO)C1(O)CC1)NC(c1cc(C(C)=O)c[nH]1)=O N1(C(C(N2CCOCC2)C)=O)CCC2(CC2NC(=O)CCC2CCCCC2)C1 c1(C(=O)NC2CN(C(COCCCCC)=O)C2)ccc2c(c1)nnn2C c1(C(=O)NCC2CN(C(C(C)=C(C)C)=O)C(C)C2)cncc(F)c1C c1(CC(N2CCCC(C)C2CNC(c2cnc(O)s2)=O)=O)ccc2ncsc2c1 C12(CNC(C(C3CCC3)OC)=O)CC1CN(C(=O)CN1CCC(C(N)=O)CC1)C2 C1(OC)(OC)CC(C)(C(N2CC(CCCCNC(C34CC(C)C3C4)=O)C2)=O)C1 C1(CNC(C(C)=C(CC)C)=O)CC(NC(c2cccc(SC(C)C)c2)=O)C(O)C1 C1(NC(C2(COCC)CC2)=O)CC2CCC1N2C(c1cc(C#N)c[nH]1)=O N1(C(C2C=C(C)CS2)=O)CC2CCN(C(c3n[nH]c4c(C)cccc34)=O)CC12 N1(C(CCC(=O)NC)=O)CCC(NC(=O)Cc2ccc(C)cc2)C12CC2 C1(CNC(C=CC=CC)=O)CCCCCN1C(c1cnc(C(F)F)nc1)=O C1(C(C(=O)NCC)N(CCCc2ccoc2)C2CC2)C2CCOCC12 C(CCCCC(=O)N(C)Cc1cccc(C)c1)N(C(C(CSC)C)=O)C CC(C)(COC1CCCC1)C(=O)NCC1C2CN(C(=O)CC(O)C3CC3)CC12 Cn1nc(C(=O)NCC2CCN(C(=O)C=CC(=O)NC3CC3)CC2)c(Br)n1 c1(CCC(=O)N(C2(C(=O)NC3CC3(C)C)CC2)C)cccc(Br)c1Cl C(CC(F)F)(C(=O)NCC1CC2CCC1CC2)N(C(=O)CCc1nccs1)C c1(C(=O)Nc2c(OC)ncc(SC)c2)cccc2cc(C)ncc12 C(=O)(C(C)CC(C)(F)F)NCC(CCCC)NC(c1cccc(S(C)=O)c1)=O C12(C(=O)NCC3C(CNC(c4nc[nH]c4C(F)(F)F)=O)C3)CCC(=O)N1CCS2 c1(OC)cc(OC)cc(CN(CC(=O)N(c2cc(C)ccc2F)C)C)c1 c1(C(N2CCC(N(C(C3CCC(C)N3C(C)=O)=O)CC)C2)=O)cc(C)cc(O)c1 N1(C(c2cc(CC)on2)=O)CCC2CC12C(=O)NCc1cc(C(N)=O)no1 C1(N(C(C(C2CC2)OCC)=O)C)CC(C)(C)C1(C)C.C12CC1C(=O)NC2C CCC(CCC(=O)N(CC(O)COC)CC)NC(c1c[nH]c(=S)cn1)=O c1(NC(C(CC2CCCC2)NC(CN(CCC#C)C)=O)=O)cncc(C2CC2)c1 C1(NC(=O)CNc2ncccn2)CCN(C(=O)Cn2cncn2)CC1 N1(C(c2ccc(C)s2)=O)CCC(O)(C(C)NC(=O)CCc2nnc(C3CC3)o2)C1 c1(OC)cnc(CNC(=O)C(C2(C)CC2)NC(C2CCC(=O)C2)=O)cn1 Cc1noc(C)c1C(C)(C)C(=O)N1CC(C)(NC(C2CCCC(F)C2)=O)C1 C(=O)(C1=NN(CCO)C(=O)CC1)N1CC(NC(=O)COc2ccc(F)c(F)c2)C1 c1(C(=O)Nc2ccc(C(=O)NCC3COC3)cn2)cc(Cl)c(Cl)cc1Cl c1(OC)cccc2c1CN(C(C1CC1c1cccc(-c3ccoc3)c1)=O)C2 CCCC(C)CC(=O)N1CCOC(CN(C)C(c2cc(CC)n(C)n2)=O)C1 C1(NC(=O)Cc2csnn2)CC(O)CN(C(=O)CCCc2ccc(Cl)cc2)C1 N1(C(COCC)=O)CCCC(O)(CNC(C2(C)COC(=O)C2)=O)C1 c1(CC(=O)N(CCCC(C)O)C)ccc(-c2ccncc2F)c(F)c1 N1(C(C(C)Oc2ccccc2)=O)CC2CCC1C2NC(=O)CC(C)C(F)F c1(C(N2CC(OC)C(NC(c3cnn(C)c3)=O)C2)=O)ncc(N)cc1Cl c1(OC)cc(Br)ccc1C(N1CCC(O)(CO)CC1)C(=O)Nc1ccc(F)cc1 c1(OC)ccc(C)cc1C(N1CC(O)CC1C)C(=O)NCCSC c1ccc2c(c1)CCSC2Cc1nc(-c2cnc3c(c2)OCO3)no1 c1(CC(N2C(C(C)NC(C3SCCS3)=O)CCC2)=O)ccc(F)cc1F Cc1cc(C(=O)NC(C)C(C)NC(=O)C=CC2CCOCC2)cc(N)c1Cl c1(N(C2CCC(NC(=O)Cc3csnn3)CC2)C)nc(O)c2c[nH]nc2n1 N1(C(C2C(OCC)C2C)=O)CCC(F)(COC(C)=O)CC1.N12CC(C(C)C1)C2=O c1(C(=O)NC2CN(C(c3cnn(CC)c3C)=O)CC2C)n[nH]c2c1CC(C)CC2 C1(CNC(CC=C)=O)CN(C(=O)C=CC(=O)NC2CC2)CC1(C)C C1(CCNC(C2ON=C(C)C2C)=O)CCN(C(c2ccc(CO)o2)=O)CC1(F)F C(CCC(C)(C)C(=O)NC1CCCCC1CNC(=O)C(C)=CC(C)(C)C)OC N1(C(CSc2ccc(C(=O)NC(C)(CO)C3CCOC3)o2)=O)CCCOCC1 N1(C(CCCCC)=O)CCC(C2CCCN(C(=O)C(C)(C)C(C)(F)F)C2)C1 C1(CC#C)CN(C(c2c(C)c(OCC)nn2C)=O)CCC1C(=O)OC(C)(C)C c1(C(=O)NC(CCOC)CNC(c2cc(Br)n[nH]2)=O)nc(O)[nH]c(=O)n1 C1(=CC)CCN(C(=O)CC(C)(C)N2CCCC2)c2ccccc21 c1(CC(N2CCCC(CNC(=O)C=CCO)C2)=O)cc(Cl)ccc1Cl C1(C(=O)NCCC2CCCN(c3ccn4nccc4n3)C2)CCC2CCCCN12 c1(C(N(CC)CC2CCCN2C(c2coc(CO)n2)=O)=O)ccc(N(C)C)nc1 CCCC(C)(CC)C(=O)NCC1CCCCCN1C(c1occ(C)c1C)=O N1(C(CC(CC)C2CC2)=O)CC(NC(=O)CCc2ccc(C)cc2)CC1(C)C C1(=O)CCC(=O)NCC(C)(C2CC2)N1.C1(C(=O)NN(C(C)=O)C)CC=CCC1 Cc1ccsc1C1CC1C(=O)NC1(C)CC(NC(C2(C(F)F)CCCO2)=O)C1 CCCC(CNC(=O)C(F)=C(C)C)NC(c1nc[nH]n1)=O c1(C(=O)NCC2N(C(CS(CC)=O)=O)CCCC2)ccc2c(n1)CCCN2 C(=O)(C(F)CC(C)(C)NC(=O)C(O)CCC)N1CC(OCCCCC)C1 N1(C(C=CC(=O)NCC)=O)CCC(NC(=O)COCCCF)CC1 c1(CC)cc(NC(C2CC(O)CN2)=O)cc(O)c1 c1(C(N2CCN(C(=O)CCCC3CC3)C(C(F)(F)F)C2)=O)ncc(F)cc1F n1(CC)cc(C(=O)N(CCCO)CC(N)=O)nn1.C1(C(=O)NCCCO)(CCl)CCC1 c1(C(C(=O)NC2CC2)N(c2ccc(C)cc2)CCCC)nn(C)c(C)c1Cl c1(OC)ccc(C2(C(=O)Nc3cc(O)nc(C(F)(F)F)n3)CC2)c(C)c1 N1(C(C)=O)CCCN(C(=O)NCc2ccc(-n3cncn3)c(F)c2)CC1 C1(COC)(CNC(C2(C)CC2(C)C)=O)CCN(C(C2CCN(C)CC2)=O)C1 C1(CCNC(C2COC(=O)O2)=O)CCCN(C(=O)CCc2ccncc2)C1 c1(CC(=O)NCC2(OC)CN(C(=O)CN3CCC(CO)CC3)C2)ccc(Cl)cc1 Cc1ncccc1NC(C1CC2CC2N1C(=O)CC1CCCN(C)C1)=O c1(Cn2ccnc2)c(F)cccc1F.N12CCCCC1CC1(CC1)NC2=O c1(N2CC(C)c3c(cncn3)C2)nc2c(c(=NCc3cccc4c3CC4)[nH]1)CCC2 C1(CNC(=O)N(c2ccc(F)cc2)CC2CC2)CN2CCCCC2CO1 N12CC(CC1=O)C2.c1(CC(=O)NCCCN(S(CC)(=O)=O)C)c(C)noc1Cl c1(C(c2nnnn2CCCCCC)NC2(CC=C)CCCC2)ncccc1CC CC(C)C(C(=O)NC1CC(CNc2ccccc2)C1)NC(c1ccccc1Cl)=O c1(C(=O)NC2CC(CCNC(C3CN(C)C3)=O)C2)c(F)ccc2occc12 Cc1ncc2n1CCC(C(=O)NC1(CNC(C3CC=CCO3)=O)CCCC1)C2 C12(NC(C3CCCCN3C(c3cncc(CO)c3)=O)=O)CCN(CC1)C2 c1(C(=O)NC2CN(C(c3cc(C)[nH]n3)=O)CC2C)cc(Cl)ccc1OC(F)(F)F N1(C(C(C2CC(NC(CC(C)=C(C)C)=O)C2)F)=O)CC2(CCN(C)CC2)C1 C1(C(N(CCCN=[N+]=[N-])CCN2CC=CC2)=O)CC=CCC1.C(=O)(COC)OC c1(C(=O)Nc2ccc(SCCCCO)cc2)ccc(I)cc1 c12ccc(cc1)C(=O)N(C)C(=O)CC2.n1(C(C)CN(C)C)cc(C(C)(C)CO)nn1 c1(C(=O)NCCN(CCOC)C(C2CC2F)=O)c[nH]c2ncc(Br)cc12 N1(C(C(c2ccc(Cl)cc2)C)=O)CCN(C(c2cc(C#N)on2)=O)CC(O)C1 C(=O)(CC(C(F)(F)F)NC(=O)C(N)=O)NC1C(C)C2CCC1C2 C=CC1CN(C(=O)C(Cc2ccco2)NC(C2CC2C(C)(C)C)=O)CCO1 C(=O)(C(C)(C)CCNC(C1CC12CCOCC2)=O)Nc1ccc(N(C)C)nc1 N1(CC(=O)NC2C(C)(COC)C2)CCN(C(=O)C=Cc2ccoc2)CC1 N1(C(C2CC=C(C)CC2)=O)CCC2(CCCN(C(=O)C(C)(F)F)C2)C1 c1(C(N(C)CC2N(C(C3(C=C)CC3)=O)CCC2)=O)ccc(N)c(C(F)(F)F)c1 C1(CNC(C(=O)Nc2c(C(=O)OC)cc(Cl)cn2)=O)CCOCC12CCC2 c1(OC)ccc(C(N2CCC(N(C(C3CC4(CCC4)CO3)=O)CC)C2)=O)c(C)c1 CCCC(C(=O)OC)C(=O)NCC(C)N(C(=O)C(C)CC(N)=O)C C1(NC(C2N(C)CCCC2)=O)CC2CC(NC(=O)Cc3csnn3)C2C1 C=CC1(C(=O)Nc2cncc(F)c2)CCN(C(C2CCOC2)=O)CC1 N1(C(c2cc(COC)no2)=O)CCC(CF)(NC(=O)CCN2CCC(F)C2)C1 CCS(=O)(=O)c1cccnc1C(N1CC(NC(c2cnc(Cl)s2)=O)C(O)C1)=O C(=O)(C1COc2c(C)cccc21)NC1CC(C)(NC(CC(COC)C)=O)C1 CCC(C)(C(=O)NCCC1(CNC(c2cnc(C)s2)=O)CC1)C(F)F C=CC(C)(C)C(=O)NCCC(O)C(=O)N1CCC(F)(CO)C1 CC1CCN(C(c2cnn(C)c2N)=O)CC1CC(=O)Nc1ccc(O)c(CO)c1 n1(CC(=O)NC2(CCC(=O)OCC)CCC2)ncc(C#N)c1N C1(C(=O)NCC23CN(C(c4ncc(N)nc4)=O)C(C2)CO3)CCN2CCCC2C1 C(N=c1[nH]c(=N)[nH]c(=NCC2CCCOC2)[nH]1)c1n(C)nnc1Br Cc1cc(O)ncc1C(=O)NCC12CC1CN(C(=O)CC(C)C1CCCCC1)C2 N1(C(Cc2c(C)nn(C)c2)=O)CCCC(C)C1CNC(=O)C(C)OCC(F)(F)F N1(C(CNS(C)(=O)=O)=O)CCC2CCCN(C(=O)CCn3ccnc3)C2C1 C1(CC)CCCN(CC(N2CC(CNC(C3CN(CC(C)C)C3)=O)C(O)C2)=O)C1 N1(C(=O)COC2(C)CCC2)CCC(CO)(O)C1.Cc1cc(C(=O)NC(C)C)no1 c1(CC(=O)N)ccccc1CC#N.N1(C(C)=O)CSCC1C(=O)NCC(CO)N c1(C(C)(F)F)ccc(C(N2CC(NC(=O)CCc3ccccn3)C(O)C2)=O)cn1 C1(CNC(Cc2ccc(C)c(Cl)c2)=O)C(C2CC2)CCN1C(=O)CC1CN(C)C1 C1(C)(CC=C)CN(C(=O)C(C2CCN(C(=O)CN3CCCC3)C2)F)C1 N1(C(C2(C#N)CCC2)=O)CCC2(CCC2NC(c2snc(Cl)c2Cl)=O)CC1 c1(C(N2C(C3(NC(C4C(=C)C4)=O)CC3)CCC2)=O)ccc(-n2cccn2)c(C)c1 C1(NC(C2CC(N(C(c3c(C)csn3)=O)C)C2)=O)CCN2CCCC12 N(C1CCc2ccc(Cl)cc21)C(c1cnc2sc(C)c(C)n21)=O C12CC3(CCN(CC3)C1=O)CO2.C(CCCCC(=O)N1CCC(C#N)C1)=CC N1(C(COCC)=O)CCCCC1CCN(C(=O)CCCC1CC1)CC C1(NC(C2C(=C)CC2)=O)CC2CC(NC(c3cccnc3OC)=O)CC2C1 N1(C(C2(COC)CCC2)=O)C2CCC1C(NC(c1ccccc1C1CCC1)=O)C2 C1(C(N(CC(CC)(C)NC(=O)CSCC(F)F)C)=O)CCC2CC1CO2 c1(C(=O)O)ccc(-c2ccc(C(N3CCCC3c3cccc(O)c3)=O)cc2)cc1 CC1(C)CCN(C(=O)CCC(F)(F)F)CC1C(=O)NCCC(N)=O N(C(=NCCCCl)NC1CC(C)N(c2ccccc2)C1)C1CC(C(C)C)C1 n1(CCC(=O)NC2CCN(C(c3nc(O)n[nH]3)=O)CC2)cnc2ccccc12 C=C(C)CC(C(=O)OC)NC(C1CC1CCNCCCC1(OC)CC1)=O N1(C(C(CC)OC)=O)CC2(CCN(C(c3[nH]ccc3-c3ccccc3)=O)C2)C1 C12CN(CCN1C)C2=O.c1(CC)nc(CNC(=O)CC2(N(C)C)CC2)oc1C C1(COC)(NC(=O)C(=Cc2cccs2)C)CCCN(C(=O)C=CC2CCCO2)C1 C1(NC(Cc2n(C)ncc2Cl)=O)CC(F)CN(C(=O)C(C2CCCCC2)=O)C1 N1(C(=O)Cc2cc(CO)on2)CCC(O)(CNC(C23CCCC2C3(F)F)=O)CC1 C1(C(=O)NCC(CNC(CNS(N)(=O)=O)=O)O)CCc2nncn2C1 c1(C(N(C(c2nccn2CC)CCC)C)=O)ccc(S(C)(=O)=O)cc1Br c1(C(=O)NCCC2CCCCN2C(=O)CC2CC3CCC2O3)cncc(F)c1Cl c1(C(=O)OC(C)(C)C)cccc(C(=O)NCCc2cccnc2)c1 CC(C)CC(c1cccs1)NC(c1nnnn1C)(C)C1CC1 c1(C(N(CCCCN(C(=O)CC2CC2(Cl)Cl)C)C)=O)c(Cl)nn(C)c1Cl C12(CC(=O)NCc3nc(COC)sc3)CCC1CN(C(c1ccccc1F)=O)C2 c1(C(C)(C)O)cnc(C(N2CCC(F)(CNC(=O)C=CCF)C2)=O)nc1 C1(NC(c2c(OC(C)C)nccc2)=O)CC2(C1)CC2N=c1ccc(Br)c(CO)[nH]1 CC(C)CC(C)CC(C)C(=O)NC1CCC(CNC(=O)C(F)C(C)(C)O)C1 N1(C(CNS(CC)(=O)=O)=O)CCCC(NC(=O)CCCC2CCC2)C1C CN1CCS(=O)(=O)CC1CC(=O)NCC1CCN(C(=O)C(F)(F)CO)CC1 c1(NCC2(OC)CCCCC2)[nH]c(=NCC2CCCN2CC)nc2ncn(C)c12 C1(NC(C(CO)NC(C)=O)=O)CN(C(C2CCCCC2C2CC2)=O)CC(C)(C)C1 n1(CC(=O)NCCOCCN(C(CCCOCC)=O)C)ncc(Br)c1C C1(NC(=O)CCC2CCCN2C(=O)C(Cl)Cl)(CO)CCCCC1 C1(C(F)(F)F)(NC(C2CCCN2C(=O)CCc2ncccc2Br)C)CNC(=O)C1 N1(C(c2cc(CC)c(CC)o2)=O)CC(F)(F)CC1(C)CNC(c1csnc1Cl)=O Cc1cc(F)ccc1C(=O)NCCCC1CC1CC(C)(C)C.C1(=O)C(O)CN1 C(C)(C)(CC(=O)NC1(c2ncon2)CCC1)n1cc(C(C(C)C)OC)nn1 c1(C(=O)Nc2cnc(C)nc2)ccc(-c2ccccc2C(=O)OCC2CC2)c(C)c1 C#CC1CN(C(C2CCC(CC)O2)C(=O)NC2CCOCC2)CCN1C CN1CCOC(C(=O)NCCC2CCCN2C(c2cccc(Cl)c2)=O)C1=O C#Cc1cc(C(=O)N(CCCCNC(=O)Cc2ccco2)CC)ccc1C c1(C(N2CCC(N(CCC)C(C3CC3C)=O)CC2)=O)cc(N(C)C)ccc1N c1(C(N2CCC(F)(C(=O)NCCCC)C2)=O)cc(Cl)c(Cl)c(Cl)c1 CC1CC(C(=O)NC2CCSCC2)CN1C(=O)CCNCC(=O)NC(=O)C=CCl C1(C(=O)NCCCN(C2CCCC2)C(C2C(C)C2C)=O)CC2CCC1C2 O=S(=O)(c1cncc(Br)c1)N1CCCC(C2CCCCO2)C1 Cc1ccc(C2CC2NC(C2CCC(=O)N2C(C)C)=O)cc1 Cc1cc(CNC2CCN(C(=O)C3CC3)CC2O)c(C)c(C)c1 C1(NC(c2c(C)ncnc2)=O)CC(C2CCN(C(=O)CCCc3ccsc3)C2)C1 C1(NC(C2N(C(C)=O)CCCC2)=O)CCC(C)N(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 C1(O)(CNC(C(C=C)OC)=O)CCCN(C(C2(C)CCCCCC2)=O)C1 CCC(C)C(C(=O)NC(C)Cc1cc(C)[nH]n1)NC(c1ccc([N+](=O)[O-])o1)=O N1(C(c2c(C)cccc2)=O)CC2CC(C(=O)NCC3C4CCCC34)C(C2)C1 C1(N(C(CCOC(C)C)=O)C)CCC(NC(=O)C(F)(F)c2cscn2)C1 c1(OC)cccc2c1OCC2NC(=O)C(N1CCSCC(CO)C1)=O C1(NC(Cc2scc(C)c2)=O)CC2CN(C(=O)C(F)(F)C3(O)CCCC3)CC12 N1(C(CCCC(=O)NC)=O)CCC(N=c2nc(SC)[nH]s2)C(C)C1 c1(C(C2CCC(=O)N2)c2nnnn2C)cc2c(Br)cccc2[nH]1.C12CCCC1CN2 N1(C(c2nccc(OC)c2O)=O)CCC2CN(C(C3CCCCCC3)=O)CC2C1 C1(C(N2CC(CCC)N(C(=O)CS(C)(=O)=O)CC2)=O)CC1C1(C)CCOCC1 CC1=NOC(C)(C(=O)NCC2CCC2NC(=O)C(C)OC2CCCCCC2)C1 n1(CC)cc(C#CC(=O)N(CC(=O)C(=O)CC)C)nn1.C(C(=O)OCCO)O c1(CC(C)C)ccc(C(N2CC(CNC(=O)C(CN(C)C)N(C)C)C(C)C2)=O)cn1 C1(C(N(C)Cc2cccnc2)=O)CC2(CC2)CN1C(=O)CC1CC2(CC2)C1 c1(NCC2OC(C)(C)CN(C(C(=O)OC)=O)C2)nc(C)nc2c1CCCC2 C1(CNC(C(C)CC2CC2)=O)CC12CCN(C(=O)Cc1ccno1)CC2 c1(OCC(=O)NCc2cccc(C(C)O)c2)cccc(C#N)c1 c1(NC(=O)C(c2ccc(F)cc2)c2ccccn2)nnc2n1CCCC2 N1(C(CC(C)C)=O)CCC2CC(NC(=O)CCc3nccs3)C2C1.C1(C2CC2)C(=O)O1 N#Cc1ccc(NC(=O)C(N2CCN(C(C3CNC(=O)N3)=O)C3CC23)=O)cc1 c1(C(=O)NCCN(C(C)C)C(C2CC2c2cn[nH]c2)=O)ccc2c(c1)CC2 N1(C(c2c(CNC(c3c(C)cc(C)o3)=O)cc[nH]2)=O)CC(=O)N(C)C(C)C1 c1(CC)sccc1C(N1CC(O)(CNC(=O)C(C)(C)OC(C)C)C1)=O CC(C)(C)CC(C(=O)N1CCC(C2CC2)C1)NC(C1CCCC1)=O N1(C(C2CC(=C)C2)=O)CCCN(C(=O)C(C)Sc2cccnc2)C(CO)C1 C1(NC(CSCCCC)=O)(CNC(c2cc(Br)n[nH]2)=O)CCCC1 c1(C(=O)NCC2C(NC(CCc3cc(OC)no3)=O)C2)cccc(N)c1C Cc1nc(C(C)C)sc1C(=O)N(CCNC(=O)C(O)C(F)F)C1CC1 c1(OC)ccc(Br)cc1C(=O)NCC1(CNC(=O)Cn2ncnn2)CC1 c1(NC(NC(c2ccccc2)CC)=S)onc(-c2ccccc2)c1C(=O)OC C1(CO)(N)CCOCC1.c1(C(N(CC(C)CNC(=O)CN(C)C)C)=O)cc(O)n(C)n1 C12(CNC(c3csc(C)c3C)=O)CCC1CCN2C(C1CCCC2(CC2)C1)=O Cn1c(CC(N2CC(CNC(C3CCC(CNC(N)=O)C3)=O)C2)=O)nnc1O c1(OC)ccc(F)cc1C(N1CC(OCCNC(=O)CC(C)C(F)F)C1)=O C1(NC(C2(CC#C)CCCO2)=O)CCC(N(C(=O)Cc2ccnnc2O)C)CC1 C1(C(=O)NCC2CCSCC2)(NC(=O)C(C2CCCCC2)O)CCCCC1 C#CCCCCC(=O)N(C(c1ccccc1)CNC(=O)CC1CC(C)(C)CO1)C C1(C(=O)NCC(CCC)CCC)CC2(CCC2)CN1C(=O)CCCCNC(N)=O C1(C(=O)NC2COCC2n2cc(C3(O)COC3)nn2)(OC)CCN(C(C)=O)C1 C1(NC(c2n(CCC)ncc2)=O)CCC2CN(C(c3ccc(C)nc3)=O)CC2C1 c1(CNC(CCOCC)=O)ccc(O)cc1F.C12CCC1NC2=O c1(C(=O)NC(C(C(C)C)C)CNC(=O)CC(C)(C)C)cnn2c(Cl)cccc12 CCC(O)C(C)C(=O)NCc1cn(-c2ccccn2)nn1.C12(CC1)CCNC2 C1(C(N2CCC(F)(C(N)=O)C2)=O)CC2(CC2)CN1C(=O)C(c1ccccc1)F c1(NCCC(N2C(CCNC(CCSCC)=O)CCC2)=O)cccn2nccc12 c1(C(N2C3CN(C(CNC(=O)NC)=O)C(C3)C2)=O)cc2cccnc2s1 CC1CN(C(=O)CCC2CCC(=O)NC2=O)CC(C)N(C(=O)CC2=CCCC2)C1 c1(OC)ccc(-c2nc(CC(C)C)nn2C2CCCC2)c(O)c1CO C#CCC(CC#C)C(=O)NC(C)(CNC(=O)Cn1c([N+](=O)[O-])cnc1C)CO c1(CC(=O)NC(CC=C)CNC(C2(CC=C)CCC2)=O)c(C)nc(CC)nc1C C(CCCCNC(C1SCC=C1C)=O)NC(COC(CC)C)=O N1(C(c2cc(C(=O)OC)nn2C)=O)CCC2(C)C(C1)C2(Cl)Cl N1(C(C(C)(C)C)=O)CCN(C(c2ccc(Br)c(Cl)c2)=O)C(CC#N)C1 c1(C(N2CCC(n3cncn3)C2)C(=O)NC2CCOC2)cc2n(n1)CCCO2 c1(OCCNC(C)=O)ccc(SC(c2nc(Cl)oc2C)c2nnnn2C)cc1 Cc1cc(C(=O)NC2CCN(C(=O)CCC(C)C)C(C)C2)c(F)cc1Cl c1(COC)nocc1C(=O)NCC1CCC1NC(=O)C(F)Cc1ccccc1 c1(OC)c(Cl)nc[nH]c1=NCC1(NC(=O)CC(=O)NC2CC2)CCCC1 N1(C(c2c[nH]c(=NC)s2)=O)CC(NCc2cc(Cl)ccc2C(F)(F)F)C2(CC2)C1 C1(C(=O)NCCCC(=O)NC)CC(C)(C)CN1C(C1CC(=O)CC(=O)C1)=O C1(CC)CN(C(=O)CCSC)CCC1NC(c1cn(C)nn1)=O c1(C(N(C2CCC(NC(C(n3c(C)ncc3)C)=O)CC2)C)=O)cc([N+](=O)[O-])c[nH]1 c1(CNC(c2ccccc2C2CC2)C)nccc2occc12 c12ccccc1C(=O)NC2.C1(CCC)CCCC1C(=O)NCCCO C(=O)(C1=CC2CCC=CCCC12)NCC1N(C(C(CC)OCC)=O)CCC1 c1(CNC(C=CCC)=O)cncc(NCCO)n1 Cc1cc(C(=O)NC2CCC(N(C(=O)Cc3csc(NC(N)=O)n3)C)C2)c(C)o1 C1(CNC(c2c(CC)nc[nH]2)=O)CCC(C)N(C(c2csc(C3CC3)n2)=O)C1 C1(c2cc(OCC)c(C)cc2)CCN(N2CCN(C(=O)CO)CC2)C1 C1(NC(C(COC(C)C)NC(c2ccnc(CO)c2)=O)=O)C(=O)OCC1(C)C c1(C(=O)NC(C2CCCN2C(C2CC(CF)C2)=O)C)cc2ccncc2cc1F N1(C(CC=C)=O)CCCCC(NC(C2CN(C)CCO2)=O)C1 c1(CNC(=O)NCCC(C)c2nc[nH]n2)c(OC(F)F)cccc1Cl N1(c2cc(N(C)Cc3ccc(C4CC4)cc3)nc(C)n2)CCCCCCCCC1 Cc1ccc(C(C)NC(C2CN(C(c3cnn(C(C)C)n3)=O)CC2C)=O)cn1 C=C(C)CCCC(=O)N(C)CC1CCCC(NC(c2cc(C)n(C)c2)=O)C1 c1(C(N2CC3(C(NC(=O)CCc4cc(Cl)no4)CC3)C2)=O)csc2ccccc12 C1(NC(c2c(OCC)c[nH]n2)=O)CN(C(=O)CCCn2ccnc2)CC(F)(F)C1 c1(CC)onc(C(=O)NCC(O)CC(=O)NCC(C)(O)CO)c1C N1(C(COCCCOC)=O)CC(O)(CNC(C2CC2(F)F)=O)C1 CC1CCC(C(N2CC(CO)C(CO)C2)=O)CN1C(c1nc[nH]n1)=O N1(CCOC(C2C3C4CCC(C4)C23)=O)CCc2c(Cl)cccc2C1 N1(C(CCCSC)=O)CC2CCC(CNC(c3c(C)nn(C)c3C)=O)C2C1 N1(C(C(C)(C)NC(N)=O)=O)CCC(F)(CNC(c2cscn2)=O)CC1 n1(C(C)(C)C)cnc(C(=O)NC2CCC2NC(=O)CCCC2CCCO2)c1 c1(C(N2C(C(N3CCC(CC(C)C)C3)=O)COCC2)=O)cc2cnccc2[nH]1 CCC(CC)CC(F)C(=O)NCc1cc(C(=O)NC(C)CS(N)(=O)=O)cs1 n1(CC(C)C)cc(C(N2CCC(C(C)NC(c3cnn(CCF)c3)=O)C2)=O)cn1 c1(OC)cc(C)ccc1C(=O)NCC1(F)CC(NC(C2CNC(=O)N2)=O)C1 CCCN=c1[nH]c(=NC)[nH]c(=NCC(C2CCCC2)N(C)C)[nH]1 Cc1nn(CC(N2CCCC(CN(C(=O)CC3CCCCO3)C)C2)=O)c(=O)n1C Cc1cnc(C(N2CC(CC(=O)N(C3CCCC3C)C)C3(CC3)C2)=O)c(C)c1 C1(C#N)(C(=O)NC(C(=O)NCc2cc(COC)no2)C)CCCCC1 c1(C(=O)NCC2CC(F)(CNC(C(COC)(F)F)=O)C2)cc(OC)cc(C)n1 C(=O)(C(CNC(=O)C(C)=C(C)C)C(C)C)N1CC(N(CC)CC)C1.NCC C1(OCC)CC2CN(C(c3cccc(OC)c3)=O)Cc3cccnc3N2C1 c1(CNC(c2c(C)csc2)=O)cc(C(=O)NCc2ccoc2)ccn1 C(=O)(C(CC(C)C)c1ccccc1)N1CCC(N(C(C[SH](CC)CC)=O)C)C1 c1(NC(C2N(C(c3ncn(C)c3)=O)CC(O)C2)=O)cnc(Br)c(Cl)c1 C1(NC(c2ccn(CCOC)n2)=O)(CO)CCCN(C(=O)CCC(C)(C)OC)C1 N1(C(C)C)CC(N=c2cc[nH]cc2S(=O)(=O)NC(c2nccs2)C)CC1(C)C Cc1[nH]nc(C(=O)NCCC2(C)CCN(C(=O)Cn3cc(C4CC4)nn3)C2)c1Cl C1(C(=O)NCC(CNC(c2c(C)cn(C)n2)=O)F)CCC(C)(C)CO1 C(=O)(C1c2cnn(C)c2CN1C(=O)C=CC(C)(C)C)N1CC2CC(C)CC2C1.OCC N1(C(C(C)C2CCC2)=O)CCOC(CCNC(c2ncoc2Br)=O)C1 C(C(CO)(CO)NC(c1nccnc1N)=O)N(C(c1nc(OCC)oc1)=O)C CC1CN(C(c2cc(O)cc(=O)o2)=O)CCC1NC(c1ccn(C)n1)=O Cn1cc(C(=O)NCC2(CNC(=O)CNS(C)(=O)=O)CC2)c(C(F)F)c1 CC1CN(C(=O)C=C(Cl)Cl)CC(CCNC(c2cn(CC(N)=O)nn2)=O)O1 c1(SCC)ccccc1CC(=O)NC12CC(NC(=O)CCc3ccccn3)(C1)C2 c1(CC(=O)NCC(C)CN(C(=O)C(F)n2cccn2)C)ccsc1Br Cc1nn(C)c(C)c1OCCCCn1c(N(C)S(=O)C(C)C)nnc1C(C)C Cc1c(C(=O)N(C2CC(NC(c3nccnc3N)=O)C2)C)cnn1C C#CC1(C(=O)Nc2ccc(OC)nc2)CCN(C(c2ccc(=NC)[nH]c2)=O)CC1 N1(C(=O)NC2(CCO)CCOCC2)CCc2nc(O)[nH]c2C1 C1(CC#C)(C(=O)N(C)CCNC(C2CC2(c2cccc(Cl)c2)C)=O)CCCCC1 C1(NC(C2C(NC(C3(C(=O)NC)CCC3)=O)C2)=O)Cc2ccccc2C1OC c1(OCC(N)=O)ccc(C(=O)NC2COCC2CNC(C2CC2(F)F)=O)cc1 CC(C)C(O)C(C)C(=O)N(C(C)(C)CC(N1CCCNC(=O)C1C(C)C)=O)C N1(C(c2nocc2Br)=O)CCCC(O)(CNC(C2(n3cnnn3)CC2)=O)C1 C1(NC(c2cccc(-c3ncon3)c2)=O)CCCCN(C(=O)Cc2nccs2)C1 Cc1ccnc(C(=O)NC(CC(=O)N2CC3CCC(C2)O3)C(F)F)c1F C(c1ccc(F)cc1)=C(C)C(N1CC2CC1C2CNC(C1CCS1(=O)=O)=O)=O c1(C(C(=O)NCCCCC(C)NC(c2c(CC)csc2)=O)=O)ccc(F)c(C)c1 C1(C(=O)NC2(CCC(=O)NCC3(C)ON=C(C)C3)CCCC2)CCC2(CCC2)C1 c1(NC(N(C)Cc2cnc(C3(C)CC3)s2)=O)ccc(-c2ncc[nH]2)nc1 C1(NC(=O)CC2CC(F)(F)C2)CCCN(C(C2(CO)CC(F)(F)C2)=O)C1 Cc1ccc(Br)c(CNC(C)(C)CO)c1.N1(C)CCC2(CC2C(=O)N)C1 c1(C(=O)NCCCCC(C)NC(C(CC)OC)=O)c(C(F)F)nc2n1CCCC2 c1(CC(N2CCC(N(CCO)C(C3(CO)COC3)=O)C2)=O)ccc2ccccc2c1 O=C1COc2c(O)cc(C(=O)NCCc3nc4ccccc4s3)cc2N1 c1(C(N2C3CN(C(=O)C4=CCCCO4)CC2CC3)=O)cc2c(O)c(Cl)ccc2[nH]1 N1(C(C2(CC(C)C)CCNC2=O)=O)CCC(NC(=O)C=Cc2ccco2)C(O)C1 CC1(C)C2CCC(C2)C1(C)CNC(c1cc(P(C)(C)=O)cs1)=O n1(CCC)cc(Cl)c(C(=O)NCC(C(C)C)Nc2ncc(C(F)F)cn2)n1 C1(O)(C(C)NC(C2(CCF)CC2)=O)CCN(C(c2scnc2Cl)=O)CC1 N1(C(N2CC(CCn3ccccc3=O)C2)=O)CCC(CC2CCCO2)CC1 C1(N(C(C(Cc2cnc[nH]2)NC(CCOCCC)=O)=O)C)CC2CCC1CC2 CCCCC(CNC(c1ccc(C(O)CF)cc1)=O)NC(c1occc1C)=O C1(NC(=O)Cc2ccc(Cl)c(F)c2)CCN(Cc2cccc(O)c2O)CC1F N1(C(COCC(C)C)=O)CCN(C(=O)C2=CCCOCC2)C(CC(C)(C)C)C1 C1(C(=O)NCc2ncccc2F)CCN(C(C2CC2(F)Cl)=O)CC1O N1(C(c2cc(OC)n[nH]2)=O)CCCC(C(C)NC(=O)C=CC(C)=O)C1 c1(OC)cc(Cc2nc(C3CC3)no2)c(C(N2CCOCC2)=O)c(F)c1 N1(C(=O)NC2CC(C)SC2)CCn2ncc(CO)c2C1 C1(O)(C(=O)NC2CC(NC(c3c[nH]cc3C(F)(F)F)=O)C2)CCOC1 c1(SC)ccc(OCC(=O)N(C)CC2CN(C(=O)CSC(C)C)CCO2)cc1 C1(NC(CC2CC(=C)C2)=O)CN(C(=O)CCCc2ccc(Cl)cc2)CC12CCC2 N1(C(CC(n2ccc(C)n2)C)=O)CCCC(C2CC2NC(c2ccc(C)o2)=O)C1 c1(C(N2CCC(NC(C(C)CC3CC3)=O)C2C)=O)cc2ccncc2cc1F c1(C(N2CCC(OCC(F)F)C2)C(=O)NCC)ccc(Cc2nccs2)cc1 Nc1ccc(C(=O)NCC(O)CNC(=O)CNC(=O)CC(F)(F)F)nc1F N1(C(Cn2nnc(C)n2)=O)CCC(C)(C)C(NC(c2cc3n(n2)CCCO3)=O)C1 Cc1nc(C(C)C)ncc1C(=O)NC12CCCC(NC(=O)C(C)C3CCC3)(C1)C2 C(=O)(CCC1=NNC(=O)CC(F)C1)N1CCC(C(C(=O)OC)C)CC1 c1(C(N(C)CC2N(C(c3c(C)scc3)=O)CCC2)=O)cccc(C#CCO)c1 c1(NCCl)cc(C)n(CC)c1C.CCC(C)(C)C(c1nnnn1CC(F)F)N(C)C CCCC(C)(C(=O)O)NC(=O)OC(C)(C)C.c12ccnc(n1)C(=O)OC2 Cc1cc(Br)cc(C)c1CN1CCCC(CCNC(C2CCCO2)=O)C1 c1(NC2CCC(C(=O)Nc3ccc(OCC)c(C#N)c3)C2)ncc2[nH]ccc2n1 C1(C(=O)NC(Cn2cc(-c3c(OC)ccc(C)c3)nn2)C)CN2CCN1CC2C C#Cc1cc(C(N2CCC(NC(C3CCS(=O)CC3)=O)C(CO)C2)=O)ccc1Cl C(=O)(CCC(C(C)C)NC(C1CCCC(=O)C1)=O)NC(COC)C1CC1 c1(C(=O)NC2C(NC(C(C(C)C)F)=O)COCC2)nn(C)c2c1CCCC2 O=C(CC=C(Cl)Cl)NC(c1cccnc1)C(=O)NCC1CCCCS1 C1(CC)(OC)CN(N2CC=CCC3(CCOCC3)C2)C1 CC(F)(F)CCC(=O)NCCN1CCCN(C(C2(C)CNC(=O)C2)=O)CC1 S(=O)(=O)(c1ccc(C(N2CCC(C)CC2CNC(c2coc(C)c2)=O)=O)o1)NC CC(C)C(C)C(CNC(=O)COC(F)(F)F)NC(c1cc(O)nc(N(C)C)n1)=O CC(CCNC(C1CC2CC2C1)=O)N=c1cc(Cl)nc(C(F)(F)F)[nH]1 CC1CN(C(C2CCN2C(c2cnn3c2CCC3)=O)=O)C2(CC2)C(=O)N1 N1(C(CSCC#C)=O)CCN(C(c2nnsc2C)=O)CC1CCO C(=O)(CC1=CCCCC1)NCC1CCN(C(C(CC)C(C)O)=O)C12CC2 C#CC1CCCCN1C(=O)Cn1nc(C)oc1=O.C1C(COC)C(=O)N1 C12(C(N3CCC(C4OCCN(C(c5c(C)ocn5)=O)C4)C3)=O)CC1COC2(C)C C1(NC(c2cnc(CNC(COCCN(C)C)=O)nc2)=O)Cc2nccn2C1 C(=O)(NN1CCCC1C(=O)NCCc1ccco1)C1CCCC(C)CC1 C(=O)(C(O)C(C)(C)C)NC1CN(C(=O)Nc2ccc(C(C)C)cc2)CC1F N1(C(CCC2CC(OC)C2)=O)CCCC1C1CCN(C(C2CC3CC3C2)=O)C1 Cn1cnc2cccc(C(=O)NC3CCC(NC(=O)Cn4cnc(=N)[nH]4)C3)c12 Cc1ccc(Oc2cccc(NC(=O)N(C(C)C(C)C)CCC#N)c2)cc1 c1(NCC2(COc3cccc(C(C)C)c3)C(CC)C2)nccc(=NCCOC)[nH]1 N1(C(COCCOCCOC)=O)CCCCC1CNC(c1c[nH]cc1C1CC1)=O N1(C(C(C(=O)NC)(C)C)=O)CCC(F)(F)C(CNC(C2(C)CCOC2)=O)C1 c1(CC)nc(-n2cccc2)sc1C(=O)NCCCNC(C12CCC(CO1)C2)=O C12(NC(C3=C(C)CCCC3)=O)CCCC1(F)CN(C(c1cc(O)ccc1C)=O)C2 c1(CC(=O)N(CC(O)CNC(C2CSC2)=O)C)c(F)cncc1Cl C1(CNC(C(C2(O)CCC2)NC(c2cn(CC)nn2)=O)=O)C(C)(C)C1(F)F Cc1noc(C)c1Cn1cc(C)nn1.C12CCN(CC1)C(=O)N2.N1(C(=O)O)CCC1 C(=O)(C(C)(C)CCS(C)(=O)=O)NC1CC(C)(NC(C(c2ccc(F)cc2)C)=O)C1 N1(C(C2CCC(CNC(c3cnn(CCO)c3)=O)C2)=O)CC2(CCOC2=O)C1 C(=O)(CC(C)C(C)(C)C)N1C(C)CC(CNC(=O)C=Cc2ncc[nH]2)C1 n1(CC)ncc(C(=O)NC2CCC(C)(CNC(c3ccoc3Cl)=O)C2)c1C1CC1 CC1CCC(Cl)=C(C(=O)NC2CCN(C(=O)CCC3COC(C)(C)O3)CC2F)C1 c1(C(N2CC3(CN(c4nc(C)c(Br)cn4)C3)C2)=O)n[nH]c2c1CC(C)CC2 CC(C)(F)C(C)(F)CNC(C12CC(NC(C3CCCC3C(N)=O)=O)(C1)C2)=O Cc1ccc(C)c(SCC(N2CCC(C(C)NC(=O)Cc3[nH]cnc3C)C2)=O)c1 c1(C(=O)NC(CC)C(=O)NCC(CNC(N)=O)(C)F)ccc(OC)nn1 c1(OC)cn(CC(=O)NC(C)(CNC(C2CCS(=O)CC2)=O)CO)c(C)cc1=O C1(=O)CC(C)(C)CN1.CCCCC(O)CNC(=O)CCCN(C)C N1(C(C2(C)CC(F)C2)=O)CC2(C1)CN(C(c1ccc3ccnn3c1)=O)CCO2 CC(=O)CCCCCCC(=O)OC.c12cccc(n1)-c1cn(nn1)C1CN(C1)C2 C12(C(=O)NC3CC(C(N(CC=C)C4CC4)=O)C3)CC(C)(CCO1)C2 C(CS(=O)(=O)C(C)C)N(C=O)CCC1C(C)CCC1 CC1CCCC(CC(=O)NC2(CNC(=O)CC3(O)CCCOC3)CCOCC2)C1 C12(NC(CC=C)=O)CC3CCC(C1C2)N3C(c1nc(O)sc1C)=O N1(C(c2cnn(C)c2Br)=O)CC2CN(C(=O)C#CC3CC3)CC2C1 CC(CCCCNC(c1ccc(CC(N)=O)cc1)=O)NC(C1(Cl)CC12CCC2)=O c1(CSCC)cccnc1C(=O)NC1CN(C(=O)CCN2CCOC2=O)C2CC12 C(=O)(C#CC1CCOC1)N1CC(CC(=O)Nc2cncc(C)c2)CC1(C)C CC(CCO)N=c1[nH]c2c(c(=NCC3(OCCO)CCOC3)[nH]1)COCC2 c1(C(N2CCCC(C)(NC(C3CC=CCC3)=O)C2)=O)cc(F)cc(F)c1N N1(C(CCC#CC)=O)CCC2CN(C(=O)CCCN3CCCCC3)CCC12 CCC(C)C(CC(=O)NC(c1nccc(O)n1)C)NC(c1ccsn1)=O c1(C(N2CCC(n3cc(-c4ccc(C)s4)nn3)(C(=O)O)C2)=O)ccc(=O)n(C)n1 c1(C(=O)NCC(CNC(C2CC(F)C2)=O)OC)ccc(N)c(OCCO)c1 C1(NC(c2c(Cl)cn(C)n2)=O)CC2(CCCN(C(=O)CC3CCC(C)(C)C3)C2)C1 c1(C(C)NCc2cccc(OCc3cccnc3)c2)ccc(Br)cc1F C1(CC=C)(NC(c2ccnc(C)c2)=O)CCN(C(C2CC2c2ccn(C)n2)=O)C1 CCC(CO)CN=C(NCC1CC1)NC1CCN(N(C)C)CC1.C(C)=O N1(C(CCOCC)=O)CC(NC(=O)C(C(F)(F)F)OC(C)=O)CC12CCCC2 C(=O)(C(C(F)(F)F)C(F)(F)F)NCC(CCNC(=O)C(c1ccc(F)cc1)F)O Cc1nc(C2CC2)ccc1C(=O)NCC(C)(C1CC1)NC(c1ccoc1Cl)=O CCC(CC)C(C(=O)NC(C)CNC(c1ccccc1N1CCOCC1)=O)OC n1(CC(=O)N2C(C)(C)O2)ncc2cccnc12.C(=O)(C(O)(C1CC1)C1CC1)C(C)=O n1(CC)nccc1C(N1CCC(CN(C(=O)C(C)c2ccco2)C)C1)=O C1(C(=O)NC2(CCO)CN(C(=O)COC(F)F)C2)Cc2cc(F)cc(F)c2O1 c1(C(=O)Nc2cccc(NC(c3cnc(OC)s3)=O)c2)cccc(C(F)F)c1Cl N1(C(C2(C=C)CCOCC2)=O)CCN(C(=O)CC2CC(C)(C)CO2)CC(C)(C)C1 c1(C(=O)NC(C(=O)NCC2(OC)CCOC2)CC2CCOCC2)cccnc1C C1(OCC(c2ccc(-n3cnnn3)cc2)=O)CCCNS1(=O)=O Cc1cc(C(=O)N(CC(=O)NCCCCF)CC2CC2)co1 C1(CC)CCCCC1C(=O)OC.N12CCC(C1)N(C)CC2=O N1(C(C(CC=CCC)C)=O)CC(C(=O)NCC(N2CCCC2)C)C(F)(F)C1 N1(C(CCC(=O)OC)=O)CC(NC(C23CCC(CC2O)C3)=O)CC(C)C1 C(=O)(CC(C)CC(=O)NC(C)(C)C(C)CC(=O)N(C)CCn1ccnc1C)OC c1(C(N2CC(COCC)(NC(=O)CSC)C2)=O)c(C2CC2)cccc1C C1(C(N2CC(OCCOC)C2)=O)(NC(=O)CCN(C)CCO)CCN(C)C1 N1(C(C2C(CC)C2)=O)CCC(OCCN(C)NC(=O)Cc2ccc(Cl)cc2)CC1 c1(N2CC3(N(C)CC3)C2)nc(=NCC2CCCOC2C(C)(C)C)[nH]c2cc[nH]c12 C1(NC(C2CC(C)=NO2)=O)CC(C)(NC(C(C)NC(COC)=O)=O)C1 N1(C(CCC#C)=O)CCC2(COC(CNC(=O)Cc3c(C)nn(CC)c3C)C2)C1 N1(C(C(C)CC(F)(F)F)=O)CCS(=N)(=O)C2(CCC2)C1 C1(CC(=O)NC(CCN(C(CC2(CSC)CC2)=O)C)(C)C)CCCC1(F)F CC1CC=C(C(=O)NC(C(N2CCC(CO)C23CCC3)=O)C(C)(C)C)CC1 c1(N(CC(C)N(C(=O)OCCC)C)C)cc[nH]c(=NCCC(C)N2CCCC2)n1 c1(C(N2CCC(C#C)(C(=O)N(CC(O)CO)C)C2)=O)cc2ncccc2[nH]1 Cc1ncc(C(N2CCC3(CC3C(=O)Nc3cnn(C4CC4)c3)C2)=O)c(C)n1 Cn1cc2c(C(=O)NC3(CO)CN(C(=O)CCCn4cccn4)C3)cccc2n1 Cc1nc(O)nc(C)c1CC(N1CCC(CO)(NC(=O)CN2CCCC2C)C1)=O c1(C(C)=O)ccccc1N1CCOCC1.c1(C2C(=O)OC(=O)C(C)O2)ccccc1 C12(C(=O)NCC3(SCC)CC3)CC(CN(C(c3cccc(C#N)c3)=O)C1)C2 C(c1c[nH]cn1)=C(C(=O)NCCCN(C(C1N(S(C)(=O)=O)CC1)=O)CCO)F CCCC(CNC(=O)CC1CCC(=O)N1C)C(=O)N1CCC(C)(C#N)C1 CC1CCN(C(=NCCc2cccs2)NCC2CCC3CC2C3(C)C)C1 N1(C(c2n(CC)cnn2)=O)CCN(C2CN(CCCN3CCCS3(=O)=O)C2)CC1 C(=O)(C(CNC(=O)CC1C(=O)NN=C1C)CC(C)C)N(C)CC1CCN(CC)C1 n1(CC(=O)N(C)CCN(C)C(C2CC(C(F)F)C2)=O)cc(-c2ccccc2)cn1 n1(CCC)cccc1C(N1CCC(CNC(c2cc(C3CCCC3)no2)=O)C1)=O N1(C(CC#N)=O)CCCC(O)(CNC(c2c(Cl)cccc2Cl)=O)C1 C1(C(C)C)CN(C(=O)Cc2cc(O)nnc2O)CCCN1C(c1ccoc1)=O c1(NC(c2n(CCC3(C)CCCC3)nnn2)c2ccoc2)ccc2c(c1)OCO2 C1(NC(c2cccc(=O)o2)=O)CC2CCC(C1)N2C(c1ccncc1)=O c1(CC)ccc(C)cc1C(=O)NC1CC(O)CN(C(=O)C(=O)NC(C)C)C1 O=C(CC1=CCCCC1)NC(CNC(C1CCCC1(F)F)=O)C1CC1 C1(NC(c2cnc3n2CCS3)=O)CCC2CCN(C(C3CC4(CC4)CO3)=O)C1C2 C1(CC)CC(C(=O)NC(c2nncs2)C)CCN1C(=O)Cc1cncn1C C1(COC)CCCC1C(N1CC(C)(NC(c2cc(C3CCCN3C)[nH]n2)=O)C1)=O CCC(C(=O)NC1(c2ccccc2)CC1)C1CCOCC1.C12COCC1C(=O)N2 Cc1cc(C(N2CCC2CNC(c2cc(Cl)cs2)=O)=O)c(C)cn1 c1(CC)ccnc(NC(c2n[nH]c(CCC)n2)=O)c1.C12(COC1)C(C1CC1)NC2 N1(C(c2cc(C)cc(C)n2)=O)CCC2(C1)CN(C(c1csnn1)=O)CCO2 Cc1nnc2n1CC(C(=O)NC1CCCC1NC(c1ccn(C)n1)=O)C2 Cc1cc(OC(F)F)c(F)cc1Cl.c1(C(N2C3C(C3)C2)=O)cc(F)c(Br)cc1F C1(NC(=O)NCCCl)CCC2(CC1)CN(Cc1cccc([N+](=O)[O-])c1Br)C2 Cn1cc(C(F)(F)F)c(C(=O)NCCC2(O)CCN(C(c3ccccc3)=O)C2)n1 C1(C(C)=O)OCC2CCCC12.N1(C=O)CCC1(C)CC(N1CC(n2cccn2)C1)=O C(=O)(C(C#N)C(C)C)N1C(C(=O)NCCSCC#C)C=CC1 C(CC(C)C)(C(=O)NCC1CC(C(N)=O)C1)N(C(c1ccc(NC)cn1)=O)C c1(C(=O)NCC2C(NC(CCCOCCC)=O)C2)cnc(OC)nc1C N1(C(c2ccc(C(=O)OC)s2)=O)CCC2(CC2C(=O)NCC2CCN(C)CC2)C1 c1(NC2CCCC(NC(Cc3cn(CCN(C)C)nc3)=O)C2)ncnc(Cl)c1F C=CC1(C(=O)NCC(c2ccccc2)CNC(=O)C(C)CC2CC2)CCCCC1 c1(C(=O)NCC(O)C2CC2)cc2cc(Br)cnc2o1 CCC1(C(=O)NCC(c2ccc3c(c2)OCCO3)O)CCCc2ccccc21 CC(C)(C(=O)N1CCN(C(=O)CC2CCC(F)(F)CO2)C(CF)C1)C(N)=O C1(CNC(C2CCC(CC)CC2)=O)CCC2CN(C(=O)CCCC3CCC3)CC12 N1(C(C(=O)Nc2cc(CC)c(C)nc2)=O)CCN(C(=O)OC(C)(C)C)C(C)CC1C C1(CC(F)F)C(=O)NC2CCC(C2)C(=O)N1.N1(C(C)C)CC(C(N)=O)C(C)C1 CC(C)C(C(C)NC(C1(C)CC1)=O)NC(c1ccc(C(F)(F)F)cn1)=O C1(c2cn(CCOC)nn2)COCCN1C(=O)NCCCSCC(=O)O C1(NC(=O)CCSc2cccc(F)c2)CN(C(=O)C2=CCOC2)CC2CCCC12 C1(CNC(C=CCOCCOC)=O)CCC2CN(C(=O)C(C)(O)C(C)C)CC12 C1(C(=O)NCC2CCCC(CNC(C3CS(=O)(=O)C3)=O)C2)CCn2cncc2C1 c1(C(N2CCC(C(C)NC(C3CC(OC)C3)=O)C2)=O)cc(Cl)cc(Cl)c1 c1(NC(C2CCCC2C(=O)NC2CC2C2CC2)=O)cncc(Cl)c1Br Cc1nc2cccc(C(=O)C(c3ccc(C)c(C)c3)C#N)c2[nH]1 C1(c2nc(C)[nH]n2)CCCCN1C(c1c[nH]nc1C(F)F)=O N1(C(C2C(C)(CC)C2)=O)CC2(CCN(C(c3c(C)cccc3C)=O)CC2)C1 CC1CN(C(=O)COC(C)(C)C)CCC1NC(=O)C(C)(C)Br C1(C(=O)NC(CC)CNC(c2cn(CCN(C)C)nn2)=O)CCS(=O)(=O)N1C CC1(CO)CCCN1C(c1ccc(CNC(c2cnns2)=O)cn1)=O Cc1cc(F)cc(C(=O)NCC2CN(C)CCN2C(=O)COC2(C)CCC2)c1N N1(c2nnc(C(C(C)(C)C)O)n2CC(F)F)CCOCC2(CCOCC2)C1 C1(CNC(c2nc(CC)oc2)=O)CCCC2CN(C(C3C4CCC(=O)C34)=O)CC12 Cc1noc2nc(C(C)C)cc(C(=O)NC3CC3CNC(c3ccnnc3)=O)c12 Cc1nsc2ncc(C(N3CCCC(C)C3C(=O)O)=O)cc12 C1(c2nc(C(CC)CC)nn2-c2c(C)noc2C)CCC2(CCC2)O1 c12cc(nn1C)C(=O)N(CC)CCNC2=O.C1(C(=O)OC)CCC(CCO)CC1 c1(NC(=O)NCc2cn(C(c3ccc(Cl)cc3)(CC)C)nn2)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(CC)(CC)NC(c2cccc(C)c2O)=O)ccc2nonc2c1 Cc1cc(C)c(C(N2CCC(C(C)(C)C)(CNC(=O)CN3CCOC3=O)C2)=O)s1 c1(NC(c2ccc(C)s2)=O)ccc(-c2cncc(F)c2)cc1 c1(COC(C)C)nc(-c2cncnc2)n(CC2CCCO2)n1 CN1CC(NC(=O)NC(C)C(=O)O)CS1(=O)=O CC(C)(CS(C)(=O)=O)C(=O)NCC1(O)CCN(C(C2CCC2C(C)(C)C)=O)CC1 CC(C)(C)C1=NOC(CN=C(NCC(C)(C)C(N)=O)NC2CCCCC2)C1 C(=O)(C(Cc1cc[nH]n1)NC(c1cscc1OC)=O)NCCC(=O)OC CC(C)C(C(=O)NCC1CC=CC(NC(=O)CSCC(N)=O)C1)c1ccccc1 CS(C)(=O)=NC(=O)C(=O)N1CCCCC(n2cc(CCCCO)nn2)C1 N1(C(c2c(CCNC(C(CSC)O)=O)n[nH]c2)=O)CCCNC(=O)CC1 N1(C(c2c(C)nsc2)=O)CCC2(CCOCC2)C(NC(c2nnc(S)n2C)=O)C1 Cn1cnc2c(NC34CCC(CC3NC(c3cnoc3)=O)C4)nc(Cl)nc12 n1(C(C)C)ncc2c(C(=O)N(C)C)cc(Br)cc12.C123CC1CN(C2)C(=O)N(C)C3 c1(CCC(=O)N(C2CC(NC(c3ccn(C4CC4)n3)=O)C2)C)nc(O)n[nH]1 C1(C(C)(C)C)(CNC(C(C)(C)OC(C)C)=O)CCN(C(C2CCCN2C=O)=O)C1 c1(-c2cn(CCC3CN(C(c4cc(CC)sc4)=O)C3)nn2)ccc(OC)cc1 N1(C(CCOCC)=O)CCC(CN=c2[nH]nc(-c3ccccc3)o2)C(C)C1 Cc1ccc(Br)c(C(N2CC3C(C2)N3C(C2CC2c2ccccn2)=O)=O)c1 C1(NC(c2cnn(C)c2N)=O)CC2CCC(C1)N2C(C1(C#N)CCOC1)=O N1(C(C2N(C)CC2)=O)CCCC(CCNC(c2cc(C3CC3)no2)=O)C1 Cc1cc(N)cc(C(N2CCOC(CNC(=O)CC3CCCSC3)C2)=O)c1F c1(C(N2C(CCNC(C(CCC)CC)=O)COCC2)=O)n[nH]c2cc(C)ccc12 C1(C(C)(C)C)(CNC(C2CCCS2(=O)=O)=O)CCN(C(=O)COCC(F)F)C1 C1(C(=O)NCC(CNC(=O)COC2CCCC2)F)C2CCC1(c1ccncc1)C2 C1(NC(C2(C)CCC2)=O)CN(C(C2CCC(F)(F)CC2)=O)Cc2ccnn2C1 C(C(C)(C)CCCO)NC(C(CSC)(C)NC(=O)C(O)C1CCC1)=O N1(C(C(=O)N(C)CCOCCNC(=O)CC2CC(=O)NC2=O)(C)C)CCCCCC1 c1(OC)ccc(-n2cc(-c3ccc(OCc4ccccc4)cc3)nn2)nn1 c1(OC)ccc(F)c(C(=O)NC2CC(CNC(c3ccc[nH]3)=O)C2(C)C)c1 c1(C(N2CC3CN(C(c4ncccc4Br)=O)CC3C2)=O)c(F)c(F)cc(F)c1F C=CCC(C)N=c1[nH]nc(SCC(CC)CO)s1 C1(C(N2CCCC2CN(C(=O)CC2C(=O)ON=C2C)C)=O)(SC)CCOCC1 C(=O)(C(F)(CNC(c1cn2ccccc2n1)=O)C(C)C)NCCOC(CC)CC C1(NC(=O)COCC2CCCC2)CC1C1CCCN(C(c2cc(Cl)cs2)=O)C1 C(=O)(C(C)(C)C(C)NC(=O)CCCCCF)N1C(COC)COCC1 c1(C(=O)NC2CC(C)(CNC(c3cc(OC)no3)=O)C2)ncccc1Br C=C1CC(C(=O)NC(C)CC(=O)OCC2CCC2(C)C)(COC)C1 CC1CN(C(C23CCOC(C)(C2)C3)=O)CCN1C(=O)C(O)Cc1cn(C)cn1 C(=O)(C#CC1(C)CCCO1)OCc1c(OC)ccc(C)c1 c1(CC(=O)NCC2CC2NC(c2cc(CO)ccc2Cl)=O)cc(O)nnc1O C(=O)(C(C)(O)CC(F)F)NCC1CCN(C(C(=COCC)C#N)=O)CC1 c1(-n2c(-c3cccc(C(C)=O)c3)nc(C(C)O)n2)ccc2c(c1)C(=O)NCC2 CCC(C)C(O)CC(=O)N1CC=CC(NC(=O)Cc2ccc(OC)cc2C)C1 CCC(CCCCCCCC)NC(=O)CC1CCN(C(c2cnc(C)cn2)=O)C1 N1(C(c2c(C)coc2)=O)CCN(CCNC(c2cnc(C(C)(C)C)nc2)=O)CC1 c1(C(N2CCC(C)(CCNC(=O)C#CC3CCC3)C2)=O)ccnc2ccsc12 c1(C(=O)NCCC(=C)CNC(c2c(C)nsc2N)=O)cnc(N2CCCC2)nc1 c1(C(=O)NCC(O)CNC(=O)C(F)F)ccc(F)c2c1OCC2 N1(C(C2N(C)C(=O)NC2)=O)CCCC2(CCN(C(c3n[nH]c(C4CC4)n3)=O)C2)C1 N1(C(=O)NCC2CC(=O)NCCC2)CCc2c(O)noc2C1 Cc1nc(NCC2CCCCO2)cc(N(C)Cc2csc(C3CC3)n2)n1 C(=O)(C1=CCCN(C(=O)C(F)(F)C2CC2)C1)N(CC(COC)O)C C1(C(=O)NC2C3CN(C(C(C(C)C)NC(C)=O)=O)CC32)CCC(=O)N(C2CC2)C1 Cc1ccsc1Cc1nnc(N2CCCC2C2CCCOC2)s1 C1(C(N(C2CC3CC(C2)N(C(C24CC(F)(C2)C4)=O)C3)C)=O)CC(C(C)(C)C)=NO1 N1(C(CCC(=O)NCCC)=O)CCC(NC(=O)C2=NNC(C(F)(F)F)C2)CCC1 Cn1nc2ccc(Br)cc2c1CN1CC(C(=O)NC(c2ccc(F)cc2)CO)C1 CCC(Cc1cccc(C)c1)C(=O)NC(CN(C)C(C1(F)CCCCC1)=O)CC C#Cc1ccc(C(=O)NCC(C)(C(C)C)NC(C2CCS2(=O)=O)=O)cc1F c1(C(c2n(CCCC)nnn2)NCc2conc2C(C)(C)C)c(I)ncn1C c1(C(=O)NC2C(CNC(=O)CC(C3CC3)C3CC3)CCC2)ncc(Br)cc1O C1(C(C)Sc2cccc(OC)c2)CCCCN1C(=O)CNC(=O)CS.C1(N)CCC1 C1(NC(c2ncc(C)cc2C)=O)C2CC3CN(C(=O)CC4CCCN4C)C1C3C2 C(=O)(C(CC(N)=O)NC(c1ccc(C#N)cn1)=O)NC(C)Cc1ncn(C)n1 c1(C(=O)NCC(CNC(C(C)NC(=O)CC(C)(C)C)=O)F)cccc2[nH]ncc12 c1(C(N(C2CCN(C(c3sccc3Cl)=O)C2)C)=O)ncnc2ccsc12 c1(C(N(CCCN(C(COCCCC)=O)C)C)=O)cn(C)nc1-c1ccoc1 N1(C(c2ccc(CC)s2)=O)CC2CC(NC(c3c(C4CC4)noc3C)=O)C1C2 c1(OC)cc2[nH]ncc2cc1C(N1CC(C)OC(C)(C)C1)=O N1(C(C(C)n2ccnn2)=O)CCN(C(=O)C=Cc2cncn2C)CC1CCO c1(C(N2CCC(C)C(CNC(C3(CF)CC3(F)F)=O)C2)=O)cccc2ccsc12 C(=O)(N=c1cc(-c2ccc(F)cc2)[nH][nH]1)C1N(c2ccc(C)cc2)CCC1 C(C)(CCCCCO)NC(C(COC)NC(C1CCCC(O)C1)=O)=O c1(C(N(CCCCN(C(CC(CC)C)=O)C)C)=O)ccc(C(=O)OC)cc1OC CCC(CCC(=O)NCC(C)(C)C(C)(C)O)NC(c1ccnnc1)=O c1(CS(=O)(=O)NC2CCCN(c3nc(O)cc(C)n3)C2)n[nH]c2c1CCSC2 Cc1cnc(C(=O)NCC2(O)CCN(C(=O)CCN(C)CCO)C2)nc1 CCCCCCCCCC(C)n1nnnc1C(C)(C)NCC.C1CCCCCO1 C1(N(CCN(C)C)Cc2ccc(C3COC3)cc2)CCC2COC1O2 n1(CC)cnc2c(N3CCC(CCO)C3)nc(=NCCCC3CCCC3O)[nH]c12 C=C(C)C(CC(=O)NCC(C)(CNC(c1cnc(C)[nH]c1=N)=O)OC)OCC c1(C(=O)NC2C(C(=O)NCc3cc(C)ns3)CC=CC2)c[n+]([O-])c(C)cn1 C1(C(=O)NC2CCC(C(N3CC(CN=[N+]=[N-])C3)=O)C2)CC(F)C(=O)N1 c1(CN(C(c2sccc2Br)C(=O)Nc2ccccc2Cl)C)ccc(Cl)cc1F C(C(C)NC(N1CCC(c2ncc(Br)cn2)CC1)=O)(C(F)(F)F)OC CC1C(NC(=O)COCCCN(C)C)CCCN1C(C1CCOC1C(F)(F)F)=O c1(C(=O)OCC)c[nH]nc1C(=O)NC1CC(F)(CNC(c2[nH]nnc2C)=O)C1 O(NC(=O)CCc1ccccn1)CC(NCP(C)(C)=O)=O Cc1cc2n(n1)CCN(C(C1CC1C=O)=O)C2.C1(N)CCN(S(=O)(=O)C(F)(F)F)CC1 C1(NC(CCCCSC)=O)CC(C(=O)NC2(c3ccc(O)cc3)CC2)C12CCC2 C1(C(=O)NC(C)CCN(C)C(c2ccccc2SCCO)=O)CC2CCC1CC2 N1(C(c2c(NC)scn2)=O)CCC(C)(CCNC(=O)CCC23CCC(CC2)C3)C1 n1(CC(=O)NCn2cccn2)cccc1C(N(CC(C)O)CC)=O c1(OC)nc(C(=O)NC2CC3CN(C(c4ccc(F)cc4C)=O)CC23)cc(O)n1 C=Cn1cc(C(N2C(C)CCC2C)C(=O)NCc2ccccc2Br)cn1 N1CCc2nc[nH]c2C1.C(CCCCC(F)(F)F)(C(=O)OCF)N1C(C)COCC1 N(C1CCCc2occc21)C(c1c(CNC(c2ccc(F)s2)=O)cccc1)=O N1(C(C(CC(C)C)C)=O)CC2(CCCC2NC(=O)Cc2cn(C3CC3)cn2)C1 C(=O)(CC(C)C(F)(F)F)NCCCNC(c1nn(C(CC)CC)c(C)c1)=O C1(C(=O)NCC2N(C(c3cnc(OC)s3)=O)CCC2)CC(=O)NC2CCCCC12 c1(OC)cccc2c1OCCCC2NC(=O)NC(c1cccc(F)c1)CF c1(OC)ccc(C2(N(C(C(=O)NCC(F)F)c3ccsc3)C)COC2)cc1 NS(=O)(=O)C1(C(N2CCC(NC(=O)CC3COCCO3)C(F)C2)=O)CCCC1 c1(OCC(N2CCC(Nc3ccc(N)cc3)C2)=O)ccc(Cl)c(Cl)c1 C1(C(N2CCOC(CCF)C2)=O)CCCC(C)(C)C1.C12(CC1)C(C)NC2=O C(=O)(C1=CCC2CCC1N2C(c1c[nH]c(=N)s1)=O)N1CC(C)CC(C(=O)OC)C1 C1(C(=O)NC(CC#C)CO)CCCCN(C(=O)CC2CCCC2)C1 n1(CC)cc(CCOC(c2cnn(C3CC3(F)F)c2)=O)cn1 c1(CC)cccc(F)c1C(=O)NC(CNC(=O)C#CC(C)(C)C)CCOC S(=O)(=O)(c1cnn(CCF)c1)NCCC(CC#C)(C)C N1(C(C2N(CC)CC2)=O)CC2(CCCN(C(C3(C)CCCN3C)=O)C2)C1 c1(C(C)=O)ccc(C(N2CCN(C3CN(C(=O)CC4C=CCC4)C3)CC2)=O)cc1 C(=O)(CCCCCF)N1CC(NC(C(C)OCC)=O)(CC)C1 c1(C(N(CCCNC(C(CC)(C)CO)=O)C)=O)cccc2nc(O)ccc12 c1(C(N2CCC(C)(NC(C3(SCC)CC3)=O)C2)=O)c(C(C)=O)[nH]c2ccccc12 N1(C(C2CC2(F)F)=O)CC2CC(C1)N(C(C1CCc3cncn3C1)=O)C2 O(NC(=O)C(C)(C)CCCNC(=O)Cc1cccs1)C(C(=O)OC)C N1(C(CCC2CCN(C)CC2)=O)CCC(O)(CNC(=O)CN2CC(C)(C)C2)CC1 N(C)(C1CCc2cccc(Br)c21)C(C1CC(OC)CN(C(=O)OC(C)(C)C)C1)=O CCS(=O)CC(=O)N(CCC(=O)NC1CC(C(C)C)C1)CC1CC1 c1(C(=O)NC2CCN(C(c3ccc(CC)cn3)=O)C2(C)C)ccccc1[N+](=O)[O-] CN1CC(C(=O)N(CC(C)(C)CNC(c2nc(O)sc2C)=O)C)NC1=O N1(C(CC2C(C)(C)C2)=O)CC(C2CN(C(C3CC(=O)N(C(C)(C)C)C3)=O)C2)C1 N1(C(c2cnc(C)n2C)=O)CCC2C(NC(=O)C(C)C3CCCO3)C2C1 C(=O)(C1CCCc2ccccc21)NS(Sc1n2ncc(C#N)c2ncc1)(=O)=O N1(C(C)=O)CCCC(C(N2CC(CCC3CCCCC3)C(C)C2)=O)CC1 C1(C(N2CCC(F)(CNC(c3c[nH]nc3[N+](=O)[O-])=O)C2)=O)CC2CC1CC2O N1(C(c2cc(OC)n(C)n2)=O)CCN(C(c2ccoc2Br)=O)CC1C1CC1 C1(C)(NC(CNc2cccc(OC)c2)=O)CCCN(C(=O)CC2CCC3CC23)C1 C1(SC)CN(C(c2cnc(C)cn2)=O)CC1NC(=O)CSCc1cccc(C)c1 C1(C(C)NC(=O)CC2C=CCCC2)CCCN(C(=O)CC23CC(C2)C3)C1 CC1CCN(C(C2CC3(CC(NC(=O)C(CO)N(C)C)C3)C2)=O)C(C)C1 CCCCCCCCNC(=O)CC1CCCN(C(=O)NC2CCC2COC)CC1 Cc1ccc(N(CCCNC(=O)NC2CCCCC2)C2CC2)n2ncnc12 C=CCCCC(C(=O)NOCC1(C)CCC1)NC(c1cnccn1)=O c1(COC(=O)Cc2ccsc2C(F)(F)F)ccccc1-c1ccccc1 N1(C(CC)=O)CCC(NC(C2CC(N(C(=O)CCC3CC(OC)C3)C)C2)=O)CC1 CCC(C)OC.C(C(=O)NCCO)NS(C)(=O)=O.C1(C)CN(C)CCCO1 c1(OCC(=O)NC(CCNC(CNS(CC)(=O)=O)=O)C)cncc(C)n1 C12(C(=O)NCC3(NC(c4ccc(N5CCOCC5)cc4)=O)CC3)CC3CC1C2C3 CC(C)(CC(=O)NCC1CCC(NC(c2ccnnc2)=O)CC1)C1CCCCC1 CC1CCCc2ncc(C(=O)N(CCCNC(c3nncs3)=O)C)n21 c1(C(c2n(CCCC)nnn2)NC2CCSC2)sc(C(=O)OCC)cc1Br C1(NC(c2ccc(C(C)=O)[nH]2)=O)CN(C(C2C3COCC23)=O)C2(CCCC2)C1 c1(C(=O)NCC(=O)NC2(C(=O)OC)CC2)ocnc1C.C(=O)(COC)N.C1CO1 c1(CSCCC(=O)NCC2N(C(C3CC(=C)C3)=O)CC2)ccccc1 Cc1ccc(OCC(=O)NCC2CCCCN2C(c2csc(Cl)c2Cl)=O)c(F)c1 c1(C(=O)NCC2(Cn3cc(-c4c(Cl)cn(C)n4)nn3)CC2)cncc2ccsc12 CC1CC(CNC(=O)Cc2ccc(Cl)s2)CCN1C(C1(NC(N)=O)CC1)=O c1(OC)ccc(-c2cn(CC(C)(C)CNC(c3nocc3C)=O)nn2)cc1OC C(=O)(C1=Cc2ccccc2C1)NC(CC)CNC(=O)CSc1ccccc1F C(=O)(C(CC(C)(C)C)NC(C1CCC(C)(C)CC1)=O)NC(C(C)F)C C1(CNC(C2CC(CCO)C2)=O)CC2(CO1)CN(C(=O)CC1CC1)C2 CC(CN(C)C(c1cc(C(N)=O)cn1C)=O)N=c1[nH]nc(C(F)F)s1 c1(CC)cccc(C(N2CCC(NC(C(=O)OC)C(C)OC)C2)=O)c1 C1(N(C(Cn2cc(C(C)O)nn2)=O)C)CCN(C(=O)C2=NOCC2)CC12CC2 N1(C(C(C)SCC)=O)Cc2cccc(CNC(=O)C=C3CCC3)c2C1 Cc1cc2[nH]c(C(=O)NCC3CN(C(c4cnccn4)=O)CC3(C)C)cc2s1 Cc1scc(C(=O)NCCC2CCCN2C(C2CC2OC(C)(C)C)=O)c1C S(=O)(=O)(c1ccc(C(=O)O)cc1)N1CCN(C(C)(C)CN)CC1 c1(C(=O)NC2CN(C(c3cc(OCC)ncc3)=O)C(C)C2)ccc(C)c(N)c1 N1(C(CCCCOCCC=C)=O)CC2(CCC(NC(=O)CC(C)(C)SC)CC2)C1 CCCC(C)C(=O)NC1(CCNC(=O)Cc2cnn(C)c2C)CC1 C1(COC(C)C)CCCC1(C)N1CCCC1CF C1(NC(=O)C2=COCC2)CCC2(CCN(C(=O)CCOCC(F)F)CC2)C1 Cc1cnn2ccc(C(=O)NCC(C)CNC(=O)Cc3csc4nccn34)nc12 CCCCCC(F)C(=O)NCC1CCC(C(=O)NC(CC)C(F)(F)F)CC1 c1(C(=O)NC2C(NC(=O)Cn3cc([N+](=O)[O-])cn3)CC2)ccc([N+](=O)[O-])[nH]1 C1(NC(CCC2CCC(N)C2)=O)CC(C2CC2)C1 n1(CC=C)cc(C(=O)NCC2CC2NC(=O)CSc2nnc(S)s2)nn1 N1(C(c2n(CC)ccn2)=O)CCC(C)(CNC(C2(C3CCCCO3)CC2)=O)C1 CC1=C(F)CN(c2ncnc(NC3Cc4cscc4C3)c2C)CC1 Cc1ccsc1-c1ccc(Cn2ccnc2-c2nnnn2-c2ccccc2)s1 C1(NC(C(C)N(CC)CC)=O)CN(C(=O)CCC2CC2(F)F)C2CCCC12 c1(N(C(C2N(C(c3c(Cl)ccc(C)c3)=O)CC(O)C2)=O)CC)cccc2c1OCO2 C12(CNC(CCS(C)(=O)=O)=O)CN(C(=O)CC3(c4ccon4)CC3)CC1CCO2 CCC(CC(F)F)CS(=O)(=O)NCCc1ccc([N+](=O)[O-])cc1F N1(C(CCN(C(CCOCC(C)C)=O)C2CC2)=O)CCCC2CC12 N1(C(=O)OC)CCN(C(=O)C(CCF)NC(C2CCOC(C(C)C)C2)=O)CC1 CC1=C(C(=O)N2CCCOC(CCNC(=O)C(F)CC(C)C)C2)SCCO1 Cc1cc(N)ccc1C(=O)NCCNC(c1cc(O)nn1C)=O c1(N2CCC(CC(=O)O)C(F)(F)C2)ccc(Br)c(S(=O)(=O)Nc2ccccc2)n1 C1(NC(=O)CCc2nc(O)n[nH]2)CCN(C(=O)CC2CCCOC2)CC1O C1(C(=O)NC(C(C)C)CN(C)C)CC2CCC(C1)N2C(=O)CCC(C)O N1(C(c2ccn(CC)n2)=O)C(C(=O)NCCN2CCNC(=O)C2)CC2CC12 c1(CC(=O)NCC(CNC(C2CCN(C)S2(=O)=O)=O)O)n[nH]c2c1CCCC2 n1(CC(C)C)cnc(C(=O)NCC2(CCNC(C3CC(C)(F)C3)=O)CC2)n1 c1(COC)cccnc1C(N1CCCC1CCNC(c1cc(C)no1)=O)=O CC(N(C)N1CCC(F)(F)C(C#N)C1)c1cccc(N2CCOC2=O)c1 Cc1nn(C)cc1C(=O)NC(C1CCN(S(=O)(=O)CC(C)C)CC1)C c1(CNc2c(C(=O)OC)sc(C)c2)cccc2ccsc12 N1(C(N(c2ccc(CC)cc2)c2c[nH]c(=N)s2)=O)CCc2cccc(Br)c2C1 N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(C2(C)COC(C)CO2)=O)CC1C N1(C(c2cc(CN(CCC)CCC)on2)=O)CCC(c2nnc(O)o2)CC1 C(N=c1cccc(S(=O)(=O)N(C2CCC2)CC2CC2)[nH]1)C1OCCC(N(C)C)C1 N1(C(C2(C)CCOCC2)=O)CCC2CN(C(c3cccc(F)c3)=O)CC2C1 CC12CSCC1CN(C(C1COCCC1NC(c1cc(Cl)no1)=O)=O)C2 CC1(C)CN(C(=O)CCCC2CCCC2)CC1C(=O)NC1CCCC1 c1(CCN2C(C3CCN(C(C4C(CC)OCC4)=O)C3)CCC2)c(C)cccc1C C12(C(=O)NC(CC=C)CO)CC(C)(CN1C(=O)CC1(OCC)CC1)C2 c1(C(N2CCN(C(c3scc(C)c3C)=O)CC2CO)=O)coc2ccccc12 Cc1cn2cc(NC(C3CC34CN(Cc3ccc(Cl)cc3O)C4)=O)ccc2n1 c1(C(=O)NCC(C)CN(C)C(c2coc(Cl)c2)=O)nccc2ccn(C)c12 CCC(C)C(O)CC(=O)N(C(C)C(N1CCCCC1CO)=O)C1CC1 C(=O)(C1=NOC(C)(C)C1)N1CCCC(N(C(C2CS(=O)C2)=O)CC)CC1 N#Cc1ccc(C2(NC(C3(c4nc[nH]n4)CC3)=O)CCC2)cc1 CC(C)C(O)C(C)C(=O)NC(C)(C)CNC(=O)CCC1CCCO1 c1(CC(=O)NC(C)CCNC(c2cn(C)nn2)=O)ccc(Cl)c(F)c1 n1(CCC)cc(C(=O)NC2CCC(F)(CNC(c3ocnc3CC)=O)C2)c(C)n1 Cc1cc(Br)cc(Cl)c1OCC(=O)NCCC#N.C123CC(C1)(C2)C(=O)N3CCO N1(C(C(C(CC)O)C)=O)CCCC12CCN(C(=O)CC1CC(C)OC1C)CC2 c1(C(C(=O)NCCOCC)N(C)Cc2cnn(C)c2)nnc(C)s1 N1(C(C(F)=CCC)=O)CCC(CNC(=O)CSc2c(C)n[nH]c2C)C1(C)C C(CCO)(C(=O)N)N(C)C.C(CCC(C)(C)C)CCn1cc(CCCO)nn1 N1(C(C(C)Cn2ccnc2)=O)CCN(C(=O)COC2CC=CC2)CC1CCO c1(C(=O)NCCC2CC(NC(C(C(C)C)N=[N+]=[N-])=O)C2)cc2nc(Cl)ccc2o1 N1(C(Cc2c(OC)cccc2)=O)CCC(O)(CNC(C2CC3CCCC23)=O)CC1 N1(C(C(N2C(C)CCC2C)C)=O)CC(NC2CCCC(C)C2)CC(C)(C)C1 Cc1[nH]c2ccc(F)cc2c1C(N1CCN(C(=O)CC2CC23CC3)C(C)C1)=O N1(C(c2ccc(C)o2)=O)CCC2CC1CN2C(=O)COc1ccc(F)cn1 c1(C(c2n(C(C)C)nnn2)NC(C)Cc2nccn2C)c(Cl)cnc(F)c1Cl c1(C(N2CC(CNC(C3C(=C)C3)=O)C(F)(F)C2)=O)cc(C(=O)OC)cc(F)c1F C1(C(C)NC(c2ccc(C)s2)=O)CCCN(C(=O)C=CC(=O)N(C)C)C1 N1(C(c2c(C(C)C)noc2)=O)CCCCC1CCNC(C1CCN1C(C)(C)C)=O Cc1n[nH]c(C)c1CC(C)C(=O)NCC(O)CN(C)C(c1cc(F)c[nH]1)=O C#CC1CN(C(=O)CCC2CCCC2)CCN1C(=O)CCc1cnc(C2CC2)o1 Cc1csc(C=CC(=O)NCC2CCC2NC(=O)CCCCc2cnn[nH]2)n1 Cc1cnc(C(C)NC(=O)NC(c2ccc(C)s2)C(=O)C2CN(C(=O)N(C)C)C2)o1.OC C(=O)(C(C)S(C)(=O)=O)NCC1(F)CCC(CNC(c2c(C)csc2)=O)C1 c1(C(N2CC=CC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)cc2n(c(=O)c1)CCS2 N1(C(C2(OC)CCOC2)=O)CC(C2CCCCN(C(=O)CP(C)(C)=O)C2)C1 C1(C(=O)NC(C2CCN(C(CN(CCC#C)C)=O)CC2)C)CC2CCC(C1)N2C C1(C(N(C2CN(C(Cc3c(C)n[nH]c3)=O)C2)C)=O)C2CC2C2CC12 c1(SCC(=O)NCC(N(C(CSCCC)=O)C)C2CC2)nncn1C C1(OC)Cc2ccccc2N(C(c2ncccc2O)=O)C1C c1(CC)ccc(O)c(C(=O)NC(C)C(C)NC(c2cnnn2C)=O)c1 CC1CCCCC1OCCC(=O)N(C)CCN(C(=O)Cc1cccnc1O)C C1(C)(CC)CC(NC(=O)C2=CCCSC2)CN1C(C1C2(CC2)C12CC2)=O N1(C(C(CC(C)C)OC)=O)CCC2(CNC(=O)O2)C1.C12CC3(COC1C3)C(=O)N2 N1(C(CNC(C)=O)=O)CCN(C)C(C(=O)NCC2CCN(S(C)(=O)=O)C2)C1 c1(NC(C(=O)NC(C)CN(C)C2CC2)=O)ccccc1S(=O)(=O)N1CCCC1 C(c1ccc(C)cc1)=CC(=O)N(C1CCN(C(c2ccnc(OC)n2)=O)C1)CC C=C(C)CC(C(=O)NCCN1CCCOCC1)NC(c1c[nH]nc1Cl)=O CC1C(C)CCC1NC(=NC)NCC(c1ccsc1)C Cc1nc2n(n1)CC(C(N1CC(CNC(C3CC4COCC(C3)C4)=O)C1)=O)CC2 N1(C(=O)Nc2ccc(OCC)cc2)CC2CC(O)C1C2NC(c1cnsc1)=O C1(C(=O)Nc2ncc[nH]2)CC(F)CN1Cc1cccc(CO)n1 C1(C(C)NC(C(C)=C(C)C)=O)CN(C(c2cccc(Cl)c2)=O)CCO1 C1(CNC(CSCC(C)C)=O)CN2CCCCC2CN1C(c1cc(C#N)cs1)=O CCC(F)(F)CC(=O)N1CCC(OCC(=O)N(C)Cc2cnn(C)c2C)C1 C(=O)(CCS(=O)(=O)N1CC(C(=O)Nc2cc(C(C)C)ncc2Br)CC(F)C1)OC N1(C(Cc2cn(C)nc2)=O)CC(NC(=O)CCn2cccc2)CC12CCC2 c1(N2CCC(=C)CC2)nc(=NCC2CC(C)(C)CO2)[nH]c2ccsc12 Cc1nc2ccc(C(N3CCC(CO)(NC(C4CC(C)(O)C4)=O)C3)=O)cc2o1 CCCC(C)(O)C(=O)N1CCC(C(C)NC(c2cnn3ccsc23)=O)C1 C(CC(C)(C)C(=O)NC1COCCN(C(=O)C=CC2CCCCCC2)C1)SC C(C(=O)N1CCCCC1NC(C)=O)(C(C)C)NCCCOC(C)C c1(C(=O)NCc2scc(CNC(Cc3c(C)noc3)=O)n2)nsc2ccccc12 N1(C(C2(C=C)CCCC2)=O)CC=C(C(=O)NC2CC(=O)NC2=O)CC1 c1(C(=O)OC)cc(C)ccc1NCC(O)CCNC(=O)C=Cc1ccc(C)cc1 C#CC1CN(C(c2cccc(F)c2CC)=O)CCN1C(=O)Cc1nocc1CC c1(C(=O)NCC(C)CNC(=O)CSC2CC2)ccccc1N1CCCCC1 C1(N(C(C(N2CCOCC2)C)=O)CCO)CCC(NC(C2CCC=CCC2)=O)CC1 CC(CCOc1ccccc1)C(=O)N1CCCCC1CNC(N)=O N1(C(c2cc(CCC)[nH]n2)=O)CCC(C2CC(NC(c3cc(F)c[nH]3)=O)C2)CC1 CC(C)(C)CC(C(=O)N1CCNC(=O)CC1)NC(c1ccncc1Cl)=O Cc1ccc(CCC(N2CCCC(NC(=O)C3=CSCCO3)CC2)=O)cc1C N12CCC(C(C)C1)C2.c1(C(C)C)ccccc1CN(C)C C1(C(=O)NC(C2CN(C(C(C=C)(C)O)=O)C2)C)CCC(C2CCCO2)O1 c1(C(=O)NC(CNC(=O)Cn2cccn2)C2CC2)cc2cnccc2cc1F C1(C(=O)Nc2csnc2C(N)=O)(NC(C=CC(=O)OCC)=O)CC12CCC2 c1(CC(=O)N(C2CCC(NC(=O)CCC#N)C2)CC)coc2cc(OC)ccc12 c1(C(N(CC(C)NC(=O)CSC)CC)=O)cnsc1 Cc1c(C(=O)NC(C)CC(=O)N(C)Cc2ccncn2)[nH]ccc1=O c1(CC(=O)NC(=O)CO)csc(=NCCC2(CSC(C)(C)C)CC2)[nH]1 O=C(NN1CCCC1C(N1CCC2(CC(F)C2)C1)=O)N.c1nc[nH]n1 C1(NC(C(c2c(C)noc2C)C)=O)CN(C(=O)Cc2ncncc2Cl)C(C)(C)C1 Cc1ocnc1CCNC(C1CCC(n2cc(CCC3CCCOC3)nn2)C1)=O C(=O)(C1CCCc2nn(C)cc21)N1C(NC(c2cccc(OCC)c2)=O)C=CC1 c1(C(N2CCC(OC)(CNC(c3ccoc3C3CC3)=O)C2)=O)ncc(N)cc1Cl CCCCCCCCC(F)C(=O)NCC(C)NC(=O)CCc1cnc(C)nc1O c1(C(=O)NC2C(C)CN(C(=O)CC3CC(O)C34CCC4)C2)cccn2c(O)nnc12 c1(N2C(C)CC(NC(c3cnn(-c4ccncc4)c3)=O)C2)ncnc(Cl)c1F c1(C(=O)NCC2C(NC(=O)C3CC3)CC2)c(Cl)cc(-c2nn[nH]n2)cc1Cl c1(C(N2CCN(C(c3ccc(Br)c(Cl)c3F)=O)CC2)=O)cc(F)c(F)c(O)c1F CCC(C)C(=O)C(=O)NC1CC(C)(NC(c2ccc(F)c(F)c2)=O)C1 c1(CCC(=O)N(C)CCNC(c2nccnc2C(N)=O)=O)c[nH]c2ccccc12 c1(SC2C(C)N(C(=O)OC(C)(C)C)CC2)ccc([N+](=O)[O-])cc1 C1(CNC(C=C(CNC(C2OCCN(CC)C2)=O)C)=O)CC(C)(C)CCO1 N(C(=NCCC(C)C)NCC(=O)NCc1ccoc1)C1CC(CC)OCC1 N1(C(c2nc(Br)nn2C)C(=O)NC(C2CC(F)(F)C2)C)CCC2(CC1)CC(O)C2 O=C(C1=NOC2(CCCN(C(=O)C=CC3CC3)C2)C1)Nc1c(F)cccc1Br c1(OC)nn(C)c(Br)c1C(N1CCC(CNC(=O)C(C)(C2CC2)OC)C1)=O C12(NC(c3nc(C)oc3)=O)CCCN(C(c3cncc(F)c3)=O)C1C2 C1(N(C(c2cnn(CCSC)c2)=O)CC)CCN(C(c2cc(O)ncn2)=O)CC1 C(=O)(C(C(C)(C)C)NC(c1nc(C)n(C2CC2)c1C)=O)N1CC2C(CC)C2C1 n1(-c2ccn(C(C)C)n2)nc(CCN(C)C)nc1-c1ccc(CO)o1 c1(OC)nscc1C(=O)NC1CCCC1CNC(=O)Cn1cnnc1O Cc1cc(N2CCN(C(=O)C(C)CC(C)C)C(C)C2)nc(S(C)(=O)=O)n1 C(=O)(CCCCCCCCC1CC1)NC1C(NC(C(N2C(=O)CCC2=O)C)=O)C1 N1(C(CC(CCCCC)C)=O)CCC2(C=C(C(=O)NCC3(F)CCN(C)C3)C2)C1 N(C(=NCCCN1CCOC1=O)NC(CC)CC)CC(N(CC)OC)=O N1(C(c2c(C)nco2)=O)C(CNC(C2C3CCC4C(C3)CC24)=O)CC2COCC12 c1(C(=O)NCC2CN(C(C(C)C)=O)C(C)C2)cc(Cl)c(F)cc1F c1(CC)nccnc1NC(=O)CC1CN(C(=O)CCOC2CCC2)CCO1 C1(CC)CCN(C(=O)CCCC(C)C)C(C(=O)NC(C)CC2CCCO2)C1 c1(CN(C(C2(CNC(CC(=O)OCC)=O)CCCC2)=O)C)ccc(C#N)cc1 Cc1ccnc(CNC(C2(NC(=O)C(n3cc(C)cn3)C)CCSC2)=O)c1 n1(CC(=O)N(CCC(C(C)C)NC(=O)C(C)(C)CN(C)C)C)ccc(O)nc1=O Cc1scnc1-c1cn(C2COCC2NC(=O)CN(C)S(N)(=O)=O)nn1 c1(C(=O)NCC2CC2CNC(C2(C3CC3)CCC2)=O)cnc(C(F)(F)F)nc1 N1(C(CN(C)CC)=O)CCC2CCN(C(=O)Cn3ncccc3=O)CC12 c1(NCC2(NC(c3ccc(OC)s3)=O)COC2)cc(OC)ccc1OCC C1(CCC)(NC(C2CN3CCC2CC3)=O)CCCN(C(C2CC23CCCC3)=O)C1 c1(OC(CCNC(C(C)CCn2cccn2)=O)=O)cnn(C)c1C#N C=CC1CN(C(=O)CC(C)(C)N(C)C(C2CC2Cl)=O)CC1O c1(C(=O)NCC2(NC(CCOC)=O)CCCC2)cnc(O)c2cccnc12 C1(C)(C(=O)NCC(CN(C(CC2C(CC)C2(F)F)=O)C)(C)C)CCCNC1=O N1(C(c2cncc(OCC)c2)=O)CCC(CNC(=O)C(CC)=C(C)CC)C1(C)C C1(c2ccccc2)(COCCNC(=O)NCCCOCC)NC(=O)N(C)C1 c1(CC(=O)NC(CNC(C2C(OCC)C2)=O)CO)ncc(C)o1 N1(C(C23CC(OC)C2C3)=O)CCC(C(C)CNC(c2cc(C(C)C)[nH]n2)=O)CC1 CCC(CC)C(F)C(=O)NCC1CN(C(=O)CN=S(C)(C)=O)CC(C)(C)C1 O=C(CCCCCCc1cccs1)NCC1CCC(NC(=O)C2=NOCC2)C1 c1(C(=O)NCCCCCNC(c2cncc(Br)c2)=O)ncncc1Cl C(=O)(CCCCCC#N)N1C2(CNC(C(CC#C)C)=O)CC(C1)C2 c1(CN2CCC(C)(C(=O)Nc3n(CCOC)ccc3)C2)cc(C#N)ccc1[N+](=O)[O-] C1(CNC(c2cc(COC)[nH]n2)=O)CN(C(c2cnsn2)=O)C2(CCOCC2)C1 C12(C(N3C4CCC(CNC(C=CS(C)=O)=O)(C4)C3)=O)CC3CC(C(=O)N1)C2C3 C1(CNC(c2cnn3c2OCC3)=O)CCC2(CN(C(C3CC(F)C3)=O)C2)O1 C1(CC(=O)NCCN(C(CCC(=O)NCC)=O)CC(C)O)SC2=NCCN2C1=O c1(C(N2CC3OCC(NC(C4N(C)CCC4)=O)C3C2)=O)cc(Cl)cc2c1CCC2 N(C1CN(CC(C(F)(F)F)OC)CCc2ccccc21)C(=O)OC(C)(C)C C(=O)(CCCCCOC)NC1CCCN(C(CC)=O)C1 C=CCC(Cc1ccccc1)C(=O)NC1(C(=O)O)CCC1(C)C CC(C)(O)C(F)C(=O)NC1(CCCNC(C2CC(n3ccnn3)C2)=O)CC1 C1(CNC(C2(NC(C)=O)CCCC2)=O)COCCN1C(C1CC(F)(F)CS1)=O C1(NC(=O)CCN2CCCC2=O)CCC2CN(C(C3(F)CCCC3)=O)CCC2C1 N1(CC)CC(C(N2CCCCC2CC(=O)NCCCC(C)(C)OC)=O)CC1=O Cc1cnc(C(N2CCN(C(=O)C(C)C(F)F)CC2CO)=O)cc1Cl C(CCF)(C(=O)NC(c1cn(C)nc1C)C)NC(CCc1cc(C)no1)=O c1(OC)ccc(S(=O)(=O)N2CCN(CC3CC(F)(F)C3)CC2)cc1 c1(OC)cnc(C(N2CCC(NC(C34CC(F)C3C4)=O)CC2)=O)nc1 c1(N2CCN(CC)C(C)(C)C2)nc2ccc(Cl)cc2c(=NC2CCC(O)C2)[nH]1 c1(CNC(C2CCCN2c2ncc(O)cn2)=O)c(F)cc(F)c(F)c1F N1(C(C(CC#C)CC#C)=O)CCC2(CC1)CN(C(=O)CC(C)(C)C#C)CC2CO N1(C(C(n2cc(-c3ccnc(CCN)c3)nn2)C)=O)CC2(CCCC2)OCC1C N1(C(C(C2CCOCC2)OCC)=O)CCCC(c2ccccc2)CC1 C12(CNC(c3c(C(C)C)cccc3)=O)CCC1CCN2C(c1nnn(C)n1)=O O=C(C#CC1CCC1)NC1(CCC(=O)NC2C3CCCOC23)CCC1 c1(C(N2CC(F)(C(=O)NC(C(=O)OC)C3CC3)C2)=O)cccc2c1CCCC2 CC1CCN(C(=O)C=CI)CC1CN=c1[nH]nc(C2CCCC2)s1 C1(CC(=O)N(CCCCNC(C2CCN2S(C)(=O)=O)=O)C)CCCC(C)(C)O1 c1(C(=O)NCC2C(NC(CC=CCC)=O)COC2)cc(C2CC2)cc(F)c1 N1(C(c2c(C)ccnc2)=O)CCC2(CC1)CC(NC(C1CN(C)CCO1)=O)CO2 N1(C(CSCC=C)=O)CCSCC1CCNC(c1cc(CCC)[nH]n1)=O Cc1nn(CC(C)C)c(Cl)c1CNCc1ccnn1CC(C)C c1(C(C)C)nc(C(N2CC(N(C)C(C3OCCC3C(C)C)=O)C2)=O)co1 C(=O)(CCCCCCC(=O)N1CCC(NC(C23CCC2C3)=O)C(F)C1)OC n1(CC(N2C(CCNC(C3C(=C)C3)=O)CCCC2)=O)cnc([N+](=O)[O-])c1 Cc1cc(=NC(=O)C(=O)N2CC(NC(=O)C(O)CC(C)C)CC23CCC3)[nH]o1 c1(C(=O)NCCCCCCNC(C2(C)CC2(F)Cl)=O)ccnc2[nH]cnc12 C1(C2CC2)(CNC(C=C(COC)C)=O)CCN(C(=O)CN2CCOCC2=O)C1 N1(C(CCC#CC)=O)CCC2CN(C(c3cc(Cl)ccc3CC)=O)CCC2C1 c1(C(N(C2CCCN(C(c3cnn(C)c3Cl)=O)C2)CC)=O)ccc(C(F)F)nc1 Cc1ccc(C=CC(N2CC(CCCCNC(C3CC4(CC4)CO3)=O)C2)=O)cc1 N(C1CCS(=O)(=O)c2ccc(Br)cc21)C(c1n(CCOC)nnn1)(C)CSC c1(C(=O)OCC)c[nH]c(=NCCCNC(=O)CCN2CCN(C)CC2)s1 c1(C(=O)NC2C(CNC(C(n3ccc(C)n3)C)=O)CC2)csc2c(F)cccc12 c1(OC(C)C)ncc(NC(=O)CCOC(C2CC2(C)CCOCCCO)=O)cn1 c1(C(=O)NCCC(C)NC(c2ccncc2F)=O)cc2ccccc2o1 C=CC(C)(CCOC)C(=O)NC1(C(=O)NCc2ncc(C)[nH]2)CCC1 C1(C(=O)NCc2ncnn2CCF)C=CCN(C(=O)CCCn2ccnn2)C1 CC(C)(C)CCC(F)C(=O)NCCCCCCNC(c1cc2c([nH]1)CCCC2)=O c1(C(N2CC3=C(CN(C(c4ccncc4Cl)=O)C3)C2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(C(N2CC(CNC(C3(C)C(CC)CCC3)=O)C2)=O)=O)Cc2ccccc2C1 C(C(=O)NCCC1CN(C(c2cnoc2C2CCOCC2)=O)C1)(C(C)C)SCC C1(NC(=O)CCC2CC2)CC(F)(F)CC1NC(=O)CN1CCC1 N1(C(C(F)OC)=O)CC(CNC(c2cc(C3CC(F)(F)C3)[nH]n2)=O)C(C)(C)C1 c1(NCN2CCN(C(C(N3C(C)CCC3C)=O)=O)CC2)cccc2ccccc12 C1(C2=CCCCCC2)(C(N2CCC(O)(C(C)(C)CNC(C3CCC3)=O)C2)=O)CC1 N1(C(CSc2n[nH]c(=N)s2)=O)CCC2(CCC2CNC(C2CCCCO2)=O)CC1 c1(CN2C(C(c3ccc(OC)cc3)OC)CCC2)c(C)cc(C)cc1C C(CN=C(NC1CCOCC1)NC1CCC(C)(C)CC1)c1ncc(C)nc1 c1(OCC)cnc(C(N2CC(OC)C(NC(=O)CN3CC(C)(OC)C3)C2)=O)cn1 N1(C(CC(CNC(C2(C(C)=O)CC2)=O)C)=O)CCCC2(CCC2)C1 C(=O)(CC(C)C(F)F)NC(CC=CC)C(=O)NCCCCCCOC C(C)(CC(=O)NCC1(C)CC(NC(=O)CC(F)F)C1)(C(F)(F)F)N(C)C C1(C(N(CC(=O)Nc2[nH]cc(CC)c2)C2CCC2)=O)CC2(CSC2)C1 N1(C(c2ccc(CC)nc2)=O)CCN(C(C2(CC(C)C)CC2)=O)CC1CCOC C1(CCC(=O)N(C)Cc2c(C)ncs2)CCCN(C(=O)C(F)c2ccco2)C1 CC(C)(C#N)CC(=O)NCc1c[nH]nc1C(=O)NCCn1cc(C(N)=O)nn1 Cc1cc(F)ccc1C(O)C(=O)N1CCC1CNC(C1CCC(N(C)C)CC1)=O C1(N(C)CC(C(N2CCCC(CC)C2)C2(COC)CC2)=O)CC2(CCC2)C1OC Cc1ncn(C)c(=O)c1C(=O)NCC1CC(F)(CNC(C2(C#N)CC2(C)C)=O)C1 c1(CCCC(=O)NC2C(CNC(c3cc(C)[nH]c3)=O)C2)nc2ccccc2[nH]1 N1(C(C(C2CC2)OCC)=O)CCN(C)CC1CNC(=O)C(C)(C)n1cc(Cl)cn1 Cc1nsc(C)c1C(=O)NC1CC(CC(=O)NC2CCCC2CCO)C1 Cc1cc(CC(N2CCCCC(N(C)C(C34CC(C)(C3)C4)=O)C2)=O)ccc1O c1(C(=O)NC2C(NC(CCCCC(CC)C)=O)C2)cc(O)nc2ccc(F)cc12 c1(CC)c[nH]c2ncnc(N3CCC(F)C(NC(=O)C(C)(C)NS(C)(=O)=O)C3)c12 N12CCC3(CC1)CC3C2=O.c1(NC(c2cnc(C)s2)=O)cccc(O)c1Cl C12(NC(C3(C)CS(=O)(=O)C3)=O)CCCC1N(C(c1ccc[nH]1)=O)CC2 C1(C(N(C)CCOCCCNC(C2(CC(F)F)CCC2)=O)=O)CCC1(F)F C12(C(=O)NCC(C)(O)C3CC3)COCC1CN(C(=O)CCOc1cccnc1)C2 O=[N+]([O-])c1cnn(CC2CC2)c1N1CCC2(C1)CC(F)C2 N1(C(c2c(C)cc(C)cc2N)=O)CCC2CCN(C(=O)C(C)S(N)(=O)=O)C2C1 CC#CCCCC(=O)NCC1CCN(C(=O)CC(C)(C)c2ccccc2)CC1C C1(NC(CN(C(=O)CCc2ccco2)CCO)=O)CC2CC1CC21CC1 c1(CN(C(C(CC)=CC)=O)C)cnn2c1CN(C(=O)C(C)CC1CCCO1)CC2 N1(C(c2cccn(C)c2=O)=O)CC2(CC(C(N3C4CCCC3COC4)=O)CO2)C1 C1(NC(CCSCC)=O)COCC1NC(=O)C(N1CCNC1=O)C N1(C(CCCN(C(C(CC)COC)=O)C)=O)CCCC(C)(O)CC1 N1(C(C2CC(=C)C2)=O)CCN(C(c2ccnc(-c3ccoc3)c2)=O)CCC1C Cc1cc(N(C2(Cc3ccccc3)CC2)C)nc(=NCC2CCC(CO)CC2)[nH]1 CC1(C)OC2CC(C(=O)NCC(CO)NC(c3cnn(C(F)F)c3)=O)CC2O1 c1(CNC(C2CC3CC(C(=O)OC)CC32)=O)ccc2c(c1)C(C)(C)OC2 C1(O)(CCNC(C(C)SCC)=O)CCN(C(c2ccc(C)n2C)=O)C1 c1(C(N2CC(OC)C(NC(C3CCC(N(C)C)C3)=O)C2)=O)ccn2nncc2c1 C1(CNC(C(CC=C)(F)F)=O)Cc2ccccc2CN1C(=O)CCc1ccoc1 C(=O)(C(C)(C(F)(F)F)N(C)C(C)=O)NCC(C)Oc1cccc(Cl)c1.C(C)(C)(C)O C1(NC(c2[nH]cc(C)c2)=O)CCC2CC1CN2C(=O)C=Cc1ccc(F)cc1F c1(OC)cc(C(=O)NCC2CC(NC(c3cncs3)=O)C23CCC3)cc(Cl)c1 Cc1ccc(C#N)cc1C(N1CCC(C)(C)C(CNC(=O)C(=O)CCCC)C1)=O Cc1cc(Cl)ccc1OCC(N1CC2(CC(NC(=O)CCCC#N)C2)C1)=O C1(C(=O)NCCC2N(C(C3(C4(C)CC4)CC3)=O)CCOC2)CC12CCCCC2 C1(NC(c2nccc(CC)c2)=O)CC2CC1CN(C(=O)C1=CCCOC1)C2 Cn1ccc(C=CC(N2CCCCC2C(c2ccccc2)c2nn[nH]n2)=O)c1 c1(CN2CC(CC)N(S(=O)(=O)C3CC3)CC2)cc(Br)cc(F)c1F c1(CCC)ncoc1C(=O)NCC(C(C)C)NC(=O)Cn1cc(C(F)(F)F)cn1 c1(C2CCN(C(C3C(C)(C)NCC3)=O)CC2)cccc2ncccc12 N1(C(c2cc(CC)nn2C)=O)CCC2(C1)CN(C(=O)CC1(C3CC3)CC1)CCO2 Cc1cccc(O)c1NC(C1CCC=CC1NC(c1cn(C)c(C)n1)=O)=O CN(C)NC(=O)CCC(=O)NCC1CC(CNC(C2CC23CCCOC3)=O)C1 C1(CNC(c2cn(C)nn2)=O)CCCCN(C(c2c(C(F)F)cccc2F)=O)C1 Cc1ccc(F)c(NC(C2(NC(=O)COCCN(C)C)CCN(C)C2)=O)c1 O=C1c2ccccc2CCC1N1C(=O)NC(CCc2ccco2)C1=O Cc1cnc(C(N2CC(O)(C(C)NC(C3CC(C)(O)C3)=O)C2)=O)c(Br)c1 C(=O)(C1=CCCOC1)N(CCCNC(=O)Cc1ccc(C(C)(C)C)cc1)CCC C1(C(=O)NC2CN(CC)C2)CCCN(C(C2(C#N)CCC2)=O)CC1 C1(CC)CN(C(=O)CC(C)C2CC2)CCC1NC(=O)CCc1cccc(O)n1 C(=O)(CC(C)(C)C(F)F)N1CC(O)(C(C(N2CCC(OCC#C)C2)=O)F)C1 C(=O)(NNC(=O)Cc1c(F)cccc1F)N(CCCN=[N+]=[N-])CCC(=O)O c1(OC)ccccc1C1CC1C(=O)NC1CC1CNC(c1ccn(C)c1C)=O c1(C(C)=O)cc(C)n(CC(=O)NCC(CCOC)NC(c2[nH]c(C)nc2C)=O)n1 N1(CCCC(=O)N2C(Nc3cc(C)c(F)cn3)CC2)C(=O)c2ccccc2C1=O C1(C(=O)NC2C3CC(NC(c4cc(OC)ncc4)=O)CC32)COCCC1(F)F c1(NCCN(C(C(C2(C)CC2)NC(C(C)OC)=O)=O)C)ccccc1 N1(C(CCOCCOC)=O)CC2(C(=O)Nc3cnc(F)c(C)c3)CCC1CC2 c1(C(N2CC(CO)C(c3ccc(OC)cc3)C2)C(=O)NC)cccnc1C c1(OC)cc(C(=O)N(CC(O)CNC(C2(C(C)C)CC2)=O)C)c2occc2c1 C12(NC(C(CCC)c3cccc(Cl)c3)=O)CCCC1CN(C(c1cnsn1)=O)C2 c1(NC(C2CC2COc2cc(NCCO)ncc2)=O)ccc(Br)cc1C(F)(F)F N1(C(N2CCN(C)CC2)C(=O)NC(C(=O)OC)C)CCC(Cc2ccsc2)CC1 c1(NC(c2ccc(=NCc3ccc(C(F)(F)F)nc3)[nH]c2)=O)c(F)cc(Br)cc1F c1(N2CC(c3ccc(C)o3)OCC2)cccc(S(=O)(=O)N(C2CC2(C)C)C)n1 CON(CCC(=O)NCc1cc(O)cc(F)c1)C(=O)c1cc(C)nc(O)n1 N1(C(C2CCC(NC(C3CC(F)C3)=O)CC2)=O)CCn2ncnc2C1 N1(C(C2(CC#C)CCC2)=O)CCCC(O)(CCNC(c2cn(C3CC3)nn2)=O)C1 C(C(=O)NC(C(=O)NC1CSC1)C1(O)CCC1)(C(C)C)SC c1(C(=O)NCC(CNC(=O)Cc2ccno2)OC)ccc(-c2ccnn2C)s1 Cc1nc2c([nH]1)CC(C(N1CCC(CNC(C3CC4(CC4)C3)=O)C1)=O)CC2 Cc1nc(C(=O)NC2CCCC2CO)cs1.c12ccc(s1)C(=O)NC2 C1(O)(C(=O)NC2C=CC(C(=O)NCCC(=C)C)C2)CCSCC1 CC1(C)CC(NC(c2cnns2)=O)CCN(c2ncnc3c2ncn3C)C1 N1(C(c2cccnc2N2CCCC2)=O)CCOCC(F)C1 CC1=C(C)CC(C(=O)NC2CC2CNC(=O)CS(=O)(=O)N2CCN(C)CC2)CC1 C1(OC)(CNC(=O)NC2CCN(Cc3ccccc3F)C2)CCSCC1 CCC(CNC(=O)CNC1CCCCC1)(CC)C(=O)NC1CCC(C(=O)OC)C1 C1(NC(=O)NCC2CC(NC(c3c(C)scc3)=O)C2)CCCCC1C(F)(F)F N1(C(c2cnc(C)[nH]2)=O)CCCC2(CCN(C(C3CC3(C)C(C)C)=O)C2)C1 N1(CC)CCNCC1C.c12c(nnn1C)CNC2=O.C1(=O)C(C(C)C)N1 C1(C(=O)NCCn2cc(C(=O)NCC3(OC)CCC3)nn2)CCC2(CC2)O1 CC1CCN(C(=O)Cn2ncnn2)CC1CNC(C1CCC(C)(C)CC1)=O C(=O)(CC(C(F)F)NC(C1(C)CC2CC2C1)=O)N(CCCCCC=C)C n1(C(C)C)cc(C(=O)NC2CC(CCNC(=O)CC3CCCO3)C2)nn1 N1C(=NCCCC2CC2)NCCCC1C.C1(OC)CCOC1(C)C.CO C1(CNC(CSC(C)C)=O)CCN(C(C2NC(=O)OC2C)=O)CC1(F)F C1(NC(COCC#C)=O)CCC2(CC1)CC2NC(c1cc(Cl)cn1C)=O N1(C(CCCCN(C(C)C)C)=O)CC(NC(c2cn(C3CC3)nn2)=O)CC(O)C1 c1(C(=O)NC2C(CO)CCN(C(C(COC)C)=O)C2)sc2ccc(Cl)cc2c1C N1(C(c2c(C)nc(CCC)s2)=O)CC2CC(C)N(C(=O)C=Cc3ncc[nH]3)C2C1 O=C1NCCN(C2CCc3ccc(F)cc32)C1CO N1(C(CCC)=O)CCC2CN(C(=O)C(C(C)CC)OC)CC2CC1 c1(CC)ccc(C(=O)NCCC(CNC(=O)C(C)OCC(F)(F)F)OC)c(O)c1 Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)N1C2(CC2)C1.c1(C2CCCC2)ccn(C)n1 C1(OC(F)F)CCN(C(=NCC2CCC2)NCC2CCCO2)C1 N1(CCCCNC(C(=O)NC(c2cncc(C(F)F)c2)CC)=O)CCC(C)(C)CC1 CC1(C(N2CC(O)(CNC(=O)Cc3cnccc3Cl)C2)=O)CCC(=O)C1 C12(C(=O)NC3CC(C)(NC(=O)CN4C(=O)CCC4=O)C3)CC=CC(C1)OC2 O=C(C1=CCCCO1)N1CCN(C(=O)C(C2CCOCC2)O)C(C2CCCC2)C1 c1(CNC)cc(C(N2CC(C(=O)NCCCNC3CCCC3)C(C)C2)=O)ccn1 Cc1ccnc(C(=O)NC(C)C(C)(C)NC(=O)C=CC(=O)N(C)C)n1 C1(C(=O)NC2CCC(CCN)C2)(OCCN)Cc2ccccc2C1 C1(NC(Cc2c(CC)con2)=O)(CO)CCN(C(C23CCCC(CO2)C3)=O)CC1 C12(C(=O)NCC3C(C(N(C)Cc4ncc[nH]4)=O)C3)CCC(C1)C2 C(=O)(C(O)CC(C)C)N1CCC(N(C(C(CC)OC)=O)CCOC)CC1 c1(C(=O)NC2CC(CNC(=O)CCc3ccncn3)C2)cnn2c1OCCC2 C1(NC(C2C(C)C2C)=O)CCN(C(c2cn(C)nc2Br)=O)C12CCC2 c1(C(N2CC(NC(=O)C3CC3)CC3(C2)CC3)=O)ccnc2c(Br)cccc12 N1(C(c2oc(C)c(S(C)(=O)=O)c2)=O)CCC2CC(C1)CN(C(C1CC1F)=O)C2 N1(C(c2cc(C)[nH]c2C)=O)CCC(F)C(NCc2ccccc2Br)C1 C(=O)(CCCC(=O)OC)NC1(C(N2CCC(C(=O)NC)C2)=O)CC1(C)C CCC(CN(C)C(C1CC1C(N)=O)=O)NC(=O)CCn1cccc1 C(CC(C)C)(C(=O)N1CCC(F)(CO)CC1)ONC(C(CC=C)C)=O c1(C(N2CCC(NC(C(C)(Cl)Cl)=O)C(CO)C2)=O)ccn2ncnc2c1 c1(C(=O)NCC2CCCN2C(C2CC23CCC3)=O)nc[nH]c2ncc(Br)c1-2 CCCC(CCC)C(=O)NC(c1nocc1C(N1C(CO)CC1C)=O)C C1(CC)CCN(C(C2(CNC(C3(C#N)CC(=O)C3)=O)CC2)=O)CC1 CCC(COC)C(=O)NC1(C(=O)N(C2CCCC2C#N)C)CCSC1 N1(C(C(Cn2cncn2)NC(C(COCC)C)=O)=O)CCCCCC1CO N1(C(c2cc(C(=O)OC)no2)=O)CCCC(NC(=O)C(C)N(C)C)C1C c1(C2(C(=O)NC3C(NC(C=CC)=O)C3)CC2)ccc(OC(F)(F)F)cc1 C1(C(=O)NCC(=O)NC2CN(C(C3CCC3)=O)C2)CCC(C2CC2)C1.C(CO)SC O=C(CCCc1cnn[nH]1)NCC1CC1CC(=O)NCC(c1cccs1)O c1(NC(C2C(C(C)NC(C3CC(O)C3(C)C)=O)OCC2)=O)cc(Cl)cnc1O O=C(NNC(=S)Nc1ccccc1Cl)C(C(F)(F)F)Nc1ccccc1 c1(C(N2CC(C)(NC(c3cccc(N)c3Br)=O)C2)=O)cc2ccc(F)cc2o1 Cc1cc(NC(C2CCCC(NC(=O)C#CC3CC3)C2)=O)n(-c2ccncc2)n1 c12ccc(cc1O)c(=O)[nH]2.c1(CC=C)c[nH]nc1Nc1ccccc1 C(=O)(CN=c1cc[nH]cc1)NC1C2CC3C(C2)C13C(N1CCC2(CC1)CC2)=O CC1(C2CCC2)CCCN1C(=O)NC(c1ccnc(F)c1)C1CC1 c1(NC(C2CC(O)CN2Cc2ccc3c(c2)OCO3)=O)cc(Cl)cc2[nH]ccc12 CCCS(=O)(=O)CC(=O)N(C1CCCC(NC(c2ccn(C)c2C)=O)C1)C C1(C(N(C(CNC(c2nc(CCC)oc2)=O)C)C)=O)Cc2cc(F)ccc2O1 C(CS(=O)(=O)c1ccc([N+](=O)[O-])cc1)N1CCC(N2CC(C)(C)C2)CC1 CC1C(NC(=O)C2=CCCCO2)CCCN1C(=O)CC(C)C1CCCO1 c1(C(N2CC(C)(C)OC3C2COC3)=O)ncnc2cc(F)cc(F)c12 N1(C(C(C(C=C)C)C)=O)CCOC2(CCC(NC(c3cc(C)ns3)=O)CC2)C1 CCCCC(C(=O)NCC(C)(C(C)C)OCCCOCC(=O)NC(C)=O)N(C)C c1(C(CC(C)C)C(=O)NCC(CC)(CC)c2ccccn2)nc2ccccc2s1 c1(CC=C)nnc(N2CCC(C(C3CC3)N(C)C)CC2)n1CC(=C)C.C(=O)C1CC1 C#CCCC(C(=O)NC1(CO)CC(OC)C1)NC(C1OC2CCC1C2)=O N1(C(c2c(C)ncnc2C)C(=O)NCCC2CC2)CCN2CCCC2C12CCC2 N1(C(CCCCC=CC)=O)CC(C)(CNC(=O)C(O)CN(C)C)CC1(C)C N1(C(C)(C)C)CCN(C(c2cccc(C(F)(F)F)c2)C(=O)NCCC2CC2)CC1 C(=O)(N=c1ccn(CCF)[nH]1)C1(CNC(c2ccc(C(N)=O)[nH]2)=O)CC(=C)C1 N1(C(CC(CC)O)=O)CCN(C(C2CC(Cl)(Cl)C2)=O)CC1CF c1(C(=O)NC(C=C)C(=O)NC(CCC)C2CCCC2)cc2occc2[nH]1 C1(C(=O)OC)CCCC(C(=O)NC2C3CC2N(C(C2CCCC2(F)F)=O)C3)C1 C(C(=O)NCCCC(C)NC(=O)Cc1nc(C2CC2)cs1)(C(C)C)SC c1(C(=O)NC(CC)CC(=O)NC2CCOCC2)c[n+]([O-])c(C)cn1 C1(COC)CN(C(=O)COc2cccnn2)CCN1C(=O)CC(C)C1CCCC1 c1(C(N2C(C)CC(NC(c3n(C)nc(C4CCC4)c3)=O)C2)=O)c(Cl)cccc1Cl N1(C(CN(C2CCC2)C(c2ccc(C)s2)=O)=O)CCCC(CC(C)C)C1 N1(C(C(C(CC)C)O)=O)CCC(C(=O)NCC(F)(F)F)=C(F)C1 N1(C(C(C)CN(C)C)=O)CC2(CNC(=O)Cn3cnc(C(F)(F)F)c3)CC1CO2 C(=O)(CCCCCCC(=O)NC)N1CCC(CC)CC1.C1(=O)CC2(CC2)N1 c1(C(=O)NCCN(C(=O)CCC2CCCC2)CC)c[nH]nc1C1CCOC1 N1(C(c2cccc(C(C)=O)c2C)=O)CCCN(C(=O)CC)CCC1.N1CCCC1 CCC(CCC(=O)NCCC(=O)N(C)C)NC(C1CC(=O)C1(C)C)=O c1(OCC)ccc(C(=O)NC(C)(CNC(=O)CC2CC=CCC2)C(C)C)cc1Cl N1(C(CC(C)F)=O)CCCC1(C)C(=O)NCC1C(C)C1C C1(CC(=O)NC2CCC(CNC(CCC=CCC=C)=O)C2)CCCCC1O C1(CC)CN(C(c2cscc2OC)=O)CCC1NC(=O)C=CCF CCCC(C)C(=O)N1CCCC1CN(C(=O)C(C)NC(=O)CC(C)(C)C)C1CC1 [N-]=[N+]=NCCCC(=O)NCC1CCCCC1NC(C1CC(CF)C1)=O Cc1cccn(CC(N2CCN(C(c3cnn(C4CCC4)c3)=O)C(C)C2)=O)c1=O N1(C(C(C(C)C)F)=O)CCC(O)C(NC(=O)C(C)(C)C2CCOCC2)C1 S(=O)(=O)(c1cccc(F)c1)NCC1(CNC(C2CC3CCCC3C2)=O)CC1 c1(COCC(c2ccc(OC(c3nc(C)sc3)=O)cc2)=O)cc(O)cc(Cl)c1 c1(CC)ccc(C(=O)NC2(CNC(C3CCC3c3ccccc3)=O)CC2)s1 N1(C(C(C)(CO)NC(=O)CCC2CCCOC2)=O)CCN(CCO)C(=O)C1 c1(N(CCCN)C(C=CC(=O)OC)=O)ncnc2cccc([N+](=O)[O-])c12.N(C)C C(=O)(C1Cc2ccc(Cl)cc21)NC1CN(C(c2n(CC)cc(Br)c2)=O)C1 N1(C(CN2CCN(C)CC2)=O)CC2COCC(C1)C2NC(=O)C1=CCCCC1 C12(C(=O)NC3(COC)CN(C(c4cnc(C5CC5)s4)=O)C3)CCC(C1)OC2 C1(NC(c2ccc(OC)c(OC)c2)=O)CC2CCC(C1)N2C(c1cc[nH]n1)=O C1(N(C)CC)CCN(C(C2(COC)CN(C(=O)C(C)CC3CCC3)C2)=O)C1 c1(C(=O)OCC(C(C)C)OC)ccc(Br)cc1Cl C1(NC(c2cc(C)c(Cl)cc2)=O)CC2CCC1N(C(C1CCCN1C)=O)C2 c1(OC)cc(N)c(C(=O)NCC2CCCN(C(C3CCCO3)=O)C2)c(Br)c1 C1(CC)CN(C)C(=O)CN1C(C12CC(CN1C(c1cc(OC)ccn1)=O)C2)=O CN1Cc2cc(CNC(=O)CCN3Cc4ccccc4C3)ccc2C1=O N1(C(C(C)(C)C)=O)CCCC2C1CCN2Cc1ccc(F)nc1 N1(CCC)CC(C(=O)NC2CC(NC(=O)CNC(c3cnoc3C)=O)C2)CC1=O CC1=NN(C)C(=O)C1CC(=O)NCC1CC(NC(=O)CCNc2ncccn2)C1 N1(C(CCN(C(=O)C(F)C2CCCC2)C)=O)C(CO)CCC12CCC2 c1(NC(N2CCC(N(C(c3c(C)onc3)=O)C)C2)=O)ccc(C(=O)OC)cn1 C1(CNC(CN(C)C)=O)CN(C(=O)CN2CCOC2=O)CC1(F)CO c1(C(=O)NCC(CN(C(=O)CC2CCCO2)C(C)C)O)ccc(-c2ccco2)o1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC1CN(C(C(CC)C#N)=O)CC1CO C(C)(C)(CC(=O)NCC1CN(C(=O)C(F)(F)c2csc(=N)[nH]2)CC1C)OC Cc1ccc(C(=O)NC(C)CCCNC(C2(C3CCCO3)CC2)=O)c(Br)c1 c1(CCCCNC(C(C)(C)n2cc(I)cn2)=O)c[nH]c2ccccc12 C1(NC(c2c(CC)[nH]cc2)=O)CCN(C(=O)C(c2cccs2)SC)CC1 Cc1nsc(=NCC2C3CN(C(C4(C(N)=O)CC4)=O)CC23)[nH]1 n1(CC(=O)NC(C)CCCNC(=O)CCc2ccc(F)cc2)ccc([N+](=O)[O-])n1 Cc1cc(C(=O)NC2CCC(NC(c3cc4scnc4[nH]3)=O)CC2)nc(C)c1 N1(C(c2cnc(COC)s2)=O)CCCCC1C1CCCN1C(=O)C=C(C)C CCC(CC)(CO)C(=O)N1C(C(=O)NC(C)C(=O)NC2CC2)CC1C c1(CC)ccc(C)nc1N(CC)CC1CCN(C(C2CCC(F)C2)=O)CC1 N1(C(CC2CC(OCC)C2)=O)CC(NC(c2cccc(CC)c2)=O)C(C2CC2)C1 c1(C)cc(C)on1.C(=O)(C(C)OC)NCC(=O)N(CCN1CC1)CC.CCS Cc1ccc(C(C)(C)N(C)C)cc1.C12CN(CCO1)C(=O)NC2 CCC(C)C(C(=O)NCCn1cnnn1)N(C(=O)Cn1ncccc1=O)C C(=O)(C1c2ccccc2CN1C(c1ccccc1Br)=O)N(C1CC1)CC Cc1cccc(Br)c1C(C)N(C1CCCC1)C(=O)N.c1(CC2CC2)ccc(F)cc1 Cc1ccc2c(=NC(=O)C3(CNCc4scnc4C)CC3)[nH][nH]c2n1 C(=O)(C1=NOC(C)C1)N1CC(CCC)C(NC(=O)C(c2ccccc2F)(C)F)C1 C(=O)(CCN(OC)C(=O)CC1(C)CC1)NCCN(CCOC)C Cn1nc2ccccc2c1CO.N12CCC3(CC3C1)NC(=O)C13CC4CC1C3C24 C1(CNC(=O)Cc2cnoc2)CC2CC1CN2C(C1CC2C=CC1C2)=O c1(C(=O)N=c2cc(CCO)[nH][nH]2)cccc2c1CN(Cc1ccc(CO)o1)CC2 CC1=C(C(=O)NCC2CCC(C(=O)Nc3cnc(C4CC4)nc3)CC2)CCC1 CC1=C(C(=O)NC2(CNC(C3CC3F)=O)CCCC2)S(=O)(=O)CCO1 CCCC(CCC)=CC(=O)NC(CCNC(C1(N(C)C)CCCCC1)=O)C(C)C N1(CCNC(n2ccc(C)n2)=O)CCCN(C)CC1.c12cncc(n1)S2 Cc1ccn(C)c1C(=O)NCCN(C(=O)CCc1ccccc1)CCO.C1(C)CC1 N1(C(C2N(C(c3c(C)con3)=O)CC(F)(F)C2)=O)CCCC2(C=CCO2)C1 C12(CC)CCC(C(N3CCC(CNC(=O)Cc4[nH]cnc4C)CC3)=O)(CC1)CO2 c1(N(CCCN2CCCC2)C)[nH]c(=NCC2CCC23CCOCC3)nc2scnc12 c1(C(N)=O)cc(C(=O)NCCCNC(=O)C=C2CCCCC2)n[nH]1 CCCCC(C(=O)NCCC(C)C)NC(C1CCCN1C(C)=O)=O N#Cc1ccc(=NC2CCc3nc(O)sc3C2)[nH]n1 CCC(C)C(C(N)=O)NC(C1CCN(C(=O)Cc2ccn(CC)n2)CCO1)=O c1(CC(=O)NC2C(Cn3cc(CC(C=C)O)nn3)CCC2)n[nH]c2c1CCCC2 C(CCCC(CO)NC(c1ncc(Br)cc1C)=O)NC(C(C=C=C)C)=O N1(C(C)C)CCNCN(C(=O)CC(C2CC2)NC(C2CC(=O)NC2(C)C)=O)CC1 N1(C(c2[nH]c(=NC)sc2)=O)CCN(C(c2cccc[n+]2[O-])=O)C(CS(C)(=O)=O)C1 CCCC(CCCNC(=O)C(C)S(C)(=O)=O)NC(C1(OC)CCOCC1)=O C1(C(=O)NCC(C(C)C)NC(CCC(=O)OC)=O)CCC2(CCC2)CO1 C1(NC(c2c(CC)cccc2C)c2nnnn2C)CCC(F)(F)CC1(C)C N1(C(C2(C=C)CC2)=O)C2CCCC1CC(CNC(C1CCCC1C1CC1)=O)C2 C(=O)(C1=C(Cl)CCC1)NCC1(O)CCN(C(CCOC)=O)C1 C1(C(C)=O)CCc2ccccc2N(C2COCC(=O)N2CC(C)C)C1 N1(C(C(F)(F)C2(OC)CC2)=O)CC2C3CCC(C2C1)N(C(C1CCC(=O)O1)=O)C3 CC(C)C(O)C(=O)N1CCC(NC(c2cccc(C(=O)OC(C)C)n2)=O)C1 C12(C(=O)NC3CCC(N(C)C(c4ccn(C)c(=O)c4)=O)CC3)CCCC(C1)OC2 C(=O)(C1Cc2ccc(Cl)cc21)N(CCCCNC(=O)C=Cc1cn(C)cn1)C C(=O)(CC1=NNC(=O)C1)N1CCC(N(C(=O)COCCCC(C)C)CC)C1 N1(C(c2c(OC)cccc2)=O)CCOC2(CCCN(c3ncc(I)cn3)C2)C1 C1(C(=O)NCC2CN(C(C(C)Oc3cccc(CO)c3)=O)C2)OCCN(C)C1=O C(CNC(=O)CCn1ncn(C)c1=O)(C(C)C(C)C)NC(C)=O CN1C(=O)CSC1=CC(=O)NC1CC1NC(c1ccnn1CCF)=O N1(C(CCC(C)OC)=O)CCN(C(c2cc3cccc(C)c3o2)=O)CC2(CC2)C1 C(CSC)(CN=c1ccc(NC(=O)OC(C)(C)C)c[nH]1)OC C=CCC(CC(F)F)C(=O)N1CC(CNC(=O)COCC)OC(C)(C)C1 c1(C(C)NC(=O)N=c2[nH]ncn2C)nc2c(c(=NCC(C)C3CC3)[nH]1)COC2 C(CCC)(CCC)=NC(C(=O)NCCC(=O)NCCO)CCOCC N1(C(C(=O)N(C)C)=O)CCCC(F)(CNC(c2ccnn2C2CCC2)=O)C1 Cc1cn(CC(N2CC3CC(NC(C4CC4F)=O)CC2C3)=O)c2ccccc12 CC(C)C(C)CC(=O)NCCS(C)(=O)=O.C123CC1CN(C2)C(=O)CCCC31CC1 Brc1cnc(N2CCN(Cc3cccc(-c4ccccc4)c3)CC2)c(Br)c1 N1(CCC(=O)NC(C)CCN(C)C(C2(n3cccn3)CC2)=O)CCCC1=O C12CCN(C1C)C(=O)CO2.C1(CC#C)CCCN1C(=O)N(C1CC1)C1CC1 Cc1cnc(Cl)cc1NC(C1C2CC1N(C(c1cnon1)=O)C2)=O C(=O)(CCCC(CC)NC(=O)C(C)OC)NCCC=C=C C1(C(=O)NC(C2CCCC2)C#C)CCN(C(c2c[nH]c(C)c2)=O)C1 c1(C(N2CCC(OCCOC)CC2)=O)cn2ccc(-c3cnoc3)cc2n1 CN1CCCC1CCC(=O)NCCOCCC(N1CC(O)(C(F)F)C1)=O CCC(CN=c1[nH]ccn2ncc([N+](=O)[O-])c12)OC(C)(C)C N1(C(C(C)SCC)=O)CCC2(C1)CN(C(=O)CSc1ccc(OC)cc1)C2 N1(C(c2cc(C)c(C)[nH]2)=O)CCC2(CCC(NC(C3(F)CCC3)=O)C2)C1 CC1(C)CCCC(O)(C(=O)NCC2(O)CCCN(c3cc(C(N)=O)ncn3)C2)C1 C12(CC(=O)NCCCC(C)NC(C3(C(C)C)CC3)=O)COC(C)(C1)C2 N1(C(C(C)N(C)C)=O)CCCC(CCNC(=O)C=Cc2ccc(Br)o2)CC1 CC(C)(C)CCC(F)C(=O)N1CC2CN(C(c3ccn(C4CC4)n3)=O)CC(C1)O2 C1(C)(CCOC)CC(c2nnnn2C2CC(F)(F)C2)(NC2CCCS2(=O)=O)C1 c1(C(=O)NC(C(=O)NC(C2CCCCC2)C#C)CC=C)cn(C)c(=O)n1C C(c1cc(F)cc(F)c1)=CC(=O)NC1CC(NCc2ccc(OC)nc2Br)C1 Cc1ccc(F)c(C(=O)NCC2CC3CC3N2C(=O)Cc2nc([N+](=O)[O-])n[nH]2)n1 n1(C2(CC3(C(=O)NCCNC(C4CCCS4)=O)CCC3)CC2)cc(Cl)cn1 C(=O)(C1=C(C)CCOC1)NCC1ON=C(C(=O)Nc2ccc(OC)cc2C)C1 C1(F)(C(=O)NC(CN(C(=O)C(=O)Nc2ncc[nH]2)CC)C)CCOCC1 N1(CCn2c(SCCC)nnc2)CCCC(C(N2CC(C)OC(C)C2)=O)CC1 C1(C(=O)Nn2ccnc2)CCC(Oc2cccc(Cl)c2)CC1.C12CCCC1O2 C(=O)(CCC(O)C(C)(C)C)NCC12CCN(C(C3(C)CC(C)C3)=O)C1CCC2 c1(CC(=O)NC(C)C(CO)NC(=O)CCc2ccn(C)n2)ccc(O)c(Cl)c1 N1(C(C(CC)(C)C)=O)CC2(CCN(C(=O)C(C(C)C)c3cnn(C)c3)C2)C1 C(=O)(CCCC(F)(F)F)NC1(CNC(C(C)(C)c2ccno2)=O)CC1 CCC(C)(CO)C(=O)N1CCC(CCNC(c2nocc2C2CC2)=O)C1 c1(C(C(n2cc(C3CCC3)nn2)C)=O)cc2ncccn2n1 C1(C(N2C(C)C(O)CCC2)=O)C2CC(F)C(C2)N1C(c1c[nH]c(=N)s1)=O C(CC(=O)NCC1CC(F)(F)C1)(C(C)C)NC(c1c(OC)ccs1)=O C1(C(=O)NC2CC(NC(CC3(COC)CCCC3)=O)C2)C2CS(=O)(=O)CC12 C(=O)(C(O)CCn1cncn1)NCC(C)(C)Cn1cc(C(C)(C)C(N)=O)nn1 C(=O)(CCCN(C)N=O)NCC1(CNC(C(CC)(C)F)=O)CCCCC1 c1(C(N2CCC(NC(C(CC=C)(C)C)=O)C2C)=O)ncc2[nH]ncc2n1 c1(OCC(C)N(C(c2ccoc2)=O)CC)cc(C)sc1C N12CCC(CC1)CNC(=O)C1(CC1)C2=O.C1(C(=O)OC)CCC1CN(C)C n1(CC)nnnc1C(C(C)C)Nc1cnn(CC(C)(C)C)c1.C1(O)(C)CCOC1 S(=O)(=O)(c1cccs1)NC(CC(COC)NC(=O)CN(C1CCS(=O)(=O)C1)C)=O [N-]=[N+]=NCCCC(=O)NCC1CC(C(=O)NCCc2cccs2)C1 c1(C(N(C(C)CNC(=O)Cn2nnnc2C)CC)=O)cc(Cl)ns1 O=C(C1CCc2ccc(Cl)nc21)NCC1CC2(CCN(C(C3CC3F)=O)CC2)C1 C1(CC(=O)N(C(CN(C(CCOC(C)C)=O)C)C)C)CN2CCC1CC2 C(=O)(CC(O)CC(C)(C)C)N1CC(C(=O)NCCCCCCC=C)N(C)CC1 c1(C(=O)NC(C2CCN(C(=O)CCC(=O)N(C)C(C)C)C2)C)nc(=O)n(C)[nH]1 N1(C(C2CN(C(N)=O)C2)=O)CCC(NC(=O)CCSC(F)(F)F)C(O)C1 Cc1cc(C)c(C(=O)NCC2COCCN2C(C2CC(=O)N(C)C2)=O)cn1 C1(NC(c2c(CC)onc2C)=O)CCCCCN(C(C2CC3OC2C2CC32)=O)C1 O=S(=O)(c1ccc(NC2CC3(CCC3)C2O)c(Br)c1)NC1CCCCC1 c1(C(c2n(C(CC)(C)C)nnn2)NCC2(C(C)C)CC2)nn(C)cc1C(F)(F)F C(C(C)N=c1cc(C(=O)OC)nc(C(C)C)[nH]1)NC(C(CC)SC)=O CC(C)(Cc1cn(CCC(=O)N2CC(c3ncc(-c4ccccc4)[nH]3)C2)nn1)CO C(=O)(C(C)(C)C(=O)NC1CCOC(C(=O)NCCC2CC=CC2)C1)OC c1(C(=O)NCC(C)N(C(c2cnc(CCC)s2)=O)C)cccc2ccc(C)nc12 Cc1nc(C(=O)NC(C)CN(C(=O)C#CC(C)C)C)nn1-c1nc[nH]n1 n1(C(C)C)cncc1C1CCCCN1.C(=O)(C)N(C)C(N)=O C(=O)(C(C)CC(C)(C)C)N1CC2C(C(=O)NC(c3c(C)cccc3)C3CC3)(C2)C1 c1(C(=O)NC2CN(C(=O)Cn3cccn3)C3CC23)ccc(CO)nc1 C1(CCC(=O)NC2CN(C)NC2=O)CCCCN(C(=O)C(C)(C)Cl)C1 Cc1cc(=NC(C)c2csc(C(C)C)n2)[nH]c(=NCCN(C)C)[nH]1 C1(=O)C(N)(C(F)(F)F)N1.C(CS(=O)(=O)NC(C)C)NCCOC C(=O)(C(F)(F)C(O)C(C)C)NCCOCCNC(c1ccc(C)cc1C(F)(F)F)=O C1(C(=O)NCC2(CCNC(c3cc(Cl)c(Cl)[nH]3)=O)CC2)CC2(C1)CC(F)C2 N1(C(c2[nH]cc(C#N)c2)=O)CCC2(CNC(=O)COCC(F)(F)F)CCCCC12 c1(C(N2CC(C(CNC(=O)OC)C)C2)=O)ccc(C(F)F)c(Cl)c1 C(=O)(C(F)C1=CCCCC1)N1CCCC(NC(c2ccc(Cl)cn2)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CCSC1CC1)Nc1cn(CC(C)C)nc1 Cc1c(NCC2(CCO)CC2)ncnc1N1CCC(c2ccccc2)C(C)O1 C1(C(=O)NCCC(C)CCNC(C2(C#N)CC2)=O)CCCC(F)(F)CC1 CC(C)(CC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)CC(F)F C#Cc1ccnc(C(=O)NCCC(C(C)C)NC(=O)CC(C)SC)c1 c1(NC(c2n(C(CC)C)nnn2)(c2ccnn2C)C)ccc(C(C)(C)C)cc1 C1(NC(C23CCC(C)(CC2)OC3)=O)CC(C2CCN(C(=O)Cn3cnnc3)C2)C1 c1(OC)nc(C(=O)NC2CCC(CCNC(=O)COC3CCC3)C2)co1 N1(C(c2onc(C)n2)=O)CCCC(C2CN(C(=O)CN3C(C)CCC3C)C2)C1 Cc1oc(CO)cc1C(=O)NC(CNC(c1csc(C(F)(F)F)n1)=O)C1CC1 c1(C(=O)NC(C2CCN(C(C3CC(F)(F)C3)=O)C2)C)ccc(O)nn1 c1(C(=O)NCCC2N(C(CC=C)=O)CC(OC)C2)cc(Cl)cc(Cl)c1Cl N1(C(C(CCC)(C)C)=O)CCN(C(=O)CC2(C)CCCCC2)CC12CCC2 CN1C(=O)c2ccc(C(=O)NC(C)(C)CNC(C3CCCC3O)=O)cc2S1(=O)=O Cc1cc(Cl)c(C(=O)NCC2CC2NC(=O)C(O)CC(F)F)cc1Cl CCCC(C)(O)CC(=O)NCC1(C)CCCN(C(=O)CN2CCCC2C)C1 c1(C(=O)NC2C=CCCN(C(CC3(C)CC(F)(F)C3)=O)C2)cc2cccnn2c1 Cc1cc(F)sc1C(N1CC(F)CC1CNC(=O)CCC1CCCC1)=O c1(C(C(=O)NCCCN(C(C=CC)=O)C(C)C)C)cc2ccccc2o1 c1(OC)cccc2sc(C(=O)OC(C3CCC4(CC3)CC4OC)=O)cc12 C1(OC)CC(CCNC(=O)C(C)NC(=O)CC(C)(C)C)N(C(=O)C2=NOCC2)C1 C1(N(C(C(CSC)O)=O)C)CN(C(=O)Cc2ccnc(O)c2)CC12CC2 CC(C)CCCC(=O)N1CCC(C(C)COC(c2ccccc2)=O)CC1 c1(NC)ccc([N+](=O)[O-])cc1C(F)(F)F.N12CCC(C1)N(C)C(=O)C1CC1C2=O C1(CC(N2CCC(C(=O)OC)C2C)=O)CC2(C1)CN(C(=O)Cn1cc(CO)nn1)C2 c1(C(N2CC(c3c(CNC(C4CCC4)=O)nco3)C2)=O)cc2c(Cl)cccc2s1 N1(C(C(CC)=CC)=O)CCC2C(C1)CN2C(c1ccn(C2CC2(F)F)n1)=O C(c1ncccc1C)=CC(=O)N(C1CCN(C(CN(CC)CC)=O)CC1)CCO C1(CC(N2CCOC(CNC(=O)CC3CC4CCC3O4)C2)=O)CCCC(F)(F)C1 C1(NC(C(C)Cc2ccccc2)=O)CN(c2nccc(Br)n2)CC(F)(F)C1 c1(C(=O)NCCCN(C(C2CCC(CC)C2)=O)C)ccc2c(c1)CCOC2 C(=O)(CCC(C(C)C)NC(=O)NC12CCC(OC)(CC1)C2)OC N1(C(c2cc(COC)[nH]n2)=O)CCCC(C(=O)NC2(C)CC3CCC2C3)CC1 CS(=O)(=O)c1cc(C(N2CC(NC(C3CC3c3ccccc3)=O)C2)=O)ccc1F Cc1cc(C(=O)NC2CN(C(C3(C)CCCN3C)=O)C2)c2nccc(C)c2c1 Cc1nc2c(C(N3CCN(C(=O)CC(C)(C)C)C(C(C)(C)C)C3)=O)ccnc2[nH]1 c1(NC(=O)NCCC2OCC(C)(C)OC2)cc(Cl)nn2cnnc12 C1(OC)CC2(CCCC2)CCN1C(=O)CCC(=O)Nc1cccc(N)c1 CC1CCC(CNC(c2cc[nH]n2)=O)N(C(=O)C=CSc2nc[nH]n2)C1 C(=O)(C(F)(F)C(C)O)N(C1CC(CNC(c2c(C)coc2C2CC2)=O)C1)CC(C)C C1(NC(c2cc(C)sc2C)=O)CN(C(c2c(C)cccc2Cl)=O)CC1C1CC1 N1(C(CN(C)CCC(C2(C)CC(C)(C)C2)C2CCC2)=O)CCN(S(C)(=O)=O)CC1 Cc1cc(C(N2CC(C(N3CC(C)CC3C(=O)N(C)C)=O)C2)=O)cnc1C C1(CC=C)(NC(C2CC2C#N)=O)CCN(C(c2ncccc2COC)=O)CC1 N1(C(C(=O)Nc2ccc(C)cc2)C)CCN(C(=O)CC#N)C(C)C1 N1(C(C(c2cccc(OC)c2)C)=O)CCN(C(=O)C#CC2(C)COC2)CC(O)C1 C1(NC(C(C=C)(C)CC)=O)CC1C1CCN(C(=O)CCNC(=O)NC)CC1 C(CCCCCC(=O)N1CCCC1C)NC(CC(CCC)C)=O C(=O)(CS(=O)CCC(F)(F)F)NCCC1CCN(C(C(CC=CC)CC)=O)CC1 C(=O)(CS(=O)(=O)C1CC1)NCC1(F)CCN(C(Cc2cc(=N)[nH]cc2)=O)C1 Cc1oc(C(N)=O)cc1C(N1C(C(c2csc(C(=O)C3CC3)c2)=O)CCC1)=O.C(C)(C)O N1(C(CC2N(C)CCCC2)=O)Cc2ccccc2C2(CC2)C1 N1(C(C(CN(CC)CC)F)=O)CCCCC1CN(C(=O)CC(=O)N(C)C)C CC(=O)C(C)CC(C)C(=O)N1CCCC(C)(NC(C2CCC(C)CC2)=O)C1 N1(C(C#CC(C)(C)O)=O)CC2(C(N3CCSC4(CCC4)C3)=O)CC1CCO2 N1(C(CCc2c(C)nccc2)=O)CCN(C(C2CCCCC2)=O)C(CF)C1 Cc1ccoc1C(=O)NC1(CO)CN(C(=O)CCC2CC(F)(F)C2)C1 C12(C(=O)NCCCC=CC)CCN(C(=O)COC)CCC1C2 CCCS(=O)(=O)C(C)C(=O)N1CCN(C(=O)CCSC2CCCC2)CC1CCO C1(O)(C(=O)NCC2C(C(=O)NCCC3C(C)C3)CCO2)CCCCC1 C(=O)(C1=CCc2ccccc21)N(CCNC(c1c(C)nc(C2CC2)nc1S)=O)CC N1(C(CCCC)=O)CCC(CNC(=O)C(=C2CCCCC2)F)C(O)C1 C1(CNC(C2CC3(CSC3)C2)=O)CC2(CCN(C(=O)COC3COC3)CC2)CO1 c1(C(=O)NC2C(CC(=O)OCC)C2)ccc(C2=CCCC2)cc1F Cc1ccc(F)c(C(=O)NCC2CC(NC(C3CCCOCC3)=O)CC2O)c1 N#Cc1cc(F)c(CN2CC(F)(C(=O)Nc3cccc(F)c3[N+](=O)[O-])C2)c(F)c1 N1(C(=O)N(C(C(CC)C)C)C2CC2)CCCN(Cc2ccccn2)CC1 C1(CNC(=O)Cc2cscn2)CCC2(CCC2)C1NC(C1CCS(=O)CC1)=O C(=O)(C(F)C(F)(F)F)NC1CN(C(c2c(C(N(C)C)=O)cccc2)=O)C2C1C2 N1(C(C)=O)CCN(C)CC1.c12cc(on1)CNC2=O.C12CC(C1)CCNC2=O C1(C(=O)NC(C)Cn2cc(CNC(C3COCOC3)=O)nn2)CCOCC1(C)C CCC(C)(O)CNC(=O)C(CN(C)C)NC(c1cn[nH]c1)=O N1(C(C2(OCC)CCOC2)=O)CCOC(CNC(c2c[nH]cc2CC(N)=O)=O)C1 N1(C(c2c(C)cncc2)=O)CCCC(C2CCN(C(=O)CC3CC3(Cl)Cl)CC2)C1 CC(C)C(C)C(=O)NC12CC(C(=O)NC3CC(n4cncn4)C3)(C1)C2 C1(C(=O)NC2CC(=O)NC2)CN(C(=O)COc2cccc(F)c2)CC(F)(F)C1 Cc1ccc2c(c1)SC(C(N1CCCC(N(C(=O)C=C3CCCC3)C)C1)=O)C2 N1(Cc2onc(CC3CCC3)n2)CCC(N2CCCC2)C(C)C1 N1(C(CNC(C(CC)C)=O)=O)CCC(F)(C(=O)N(C2CCC2)C)CC1 C1(NC(c2cccc(CC)n2)=O)CC(O)CN(C(c2ccc(F)cc2Cl)=O)C1 c1(C(C(=O)NC(CCN(C(c2cc(C(C)=O)on2)=O)C)C)O)ccccc1Cl Cc1cc(C(N2CCOC(CNC(=O)C(F)C3CCCC3)C2)=O)nnc1C C12NC(=S)N(C3=C1C(=O)OC3)CC(CC)C1C23C(C)(C)C(CC3)C1 C1(OCCN)CCNC1.c1(C(C(=O)CCc2cnoc2)=O)cc(CCCO)on1 c1(C(N2CC(C)(COC)C2)=O)cnn2ccccc12 N1(C(CCOCCCOC)=O)CCC(CN(C(=O)CCCc2ncco2)C)C1 C1(C(=O)NC(CC)CNC(c2ccncn2)=O)CC(=O)NC(CC)C1 c1(CC)cc(C(=O)NCC2CC(NC(=O)CSS(C)(=O)=O)C23CCC3)cc(N)c1 CC1CCN(C(c2cccc(CN(C)C)c2)=O)C1CO.C(=O)(CCN)N c1(C(N2CCOC(CC3CC3)C2)C(=O)NCCCC)noc2c1CCC2 N1(C(C2CC(C#C)(O)C2)=O)C(CNC(c2n[nH]cc2Cl)=O)CC2CCCC12 N1(C(C(C)(C)SC)=O)CCCC(CCNC(=O)C(C)n2cncn2)C1 CN1CCC(C)(C(=O)NCC(C)(C)NC(=O)CC2(C#N)CC2)C1=O N1(Cc2ccc(C)cc2)Cc2ccccc2C1C(=O)NCC1CCC(F)(F)C1 c1(CC(=O)NCCN(C(C(C)OCc2ccccc2)=O)C)c(Br)cnn1C N1(C(CC(C)CF)=O)CCC2(CCCN(C(=O)CCCC(F)(F)F)C2)C1 C(=O)(C(C)(C)C)NCCCN(CC(F)(F)F)CCN(C)C c1(C(C(=O)NCC(CNC(C=C(C)C(C)C)=O)O)O)ccc(F)cc1 C1(CNC(=O)CCc2ccoc2)CCCC1NC(=O)CCc1cnco1 c1(N2CCC(CNC(C(CCC)SC)=O)C2)ncnc2c1ncn2C(C)(C)CO C1(C(N2C(C)CC(NC(CCOCC#C)=O)C2)=O)Cc2cccnc2C1 c1(CC)cc(CN(C)CC2CCCN2C(=O)CN(C(=O)C(C)OC)C)no1 C(C)(C)(CC(C)(O)COC(C)=O)NC(N1CCC(c2c(CC)cccc2)C1)=O C(=O)(C(F)CCC(C)C)N1CCN(C(c2ncc(OC)cn2)=O)CC1C CC1CCCC(C(N2CCC(NC(=O)CC3(CO)CC3)C(F)C2)=O)CC1 c1(OC2CCCC(C)C2)ccc(Br)cc1NC(=O)C(=O)NCc1ccccc1 N1(C(C(C)Oc2scc(C)n2)=O)CCC(C)C(CNC(=O)Cc2cc[nH]n2)C1 C#CC1(C)CCCN(C(C2CC(NC(=O)Cc3nccn3C)C2(C)C)=O)C1 N1(C(CN2CC(=O)N(C)C2=O)=O)CCC2(CCC2)C(CNC(C2CC2(F)F)=O)C1 C=CCCC(C(=O)N1CCC(OCCN(C)C)C1)NC(c1ccnc(F)c1F)=O N1(C(C(C)n2ccnc2)=O)CC2(CNC(=O)Cc3nc(C4CC4)n[nH]3)CC1CO2 C1(NC(c2ncncc2Cl)=O)CCC2(CCCN(C(=O)C=C3CCCCC3)C2)C1 C1(C)(CCC)CCCN(C(=O)C(C2CCC2)NC(=O)Cn2ccc(C(F)F)n2)C1 c1(CNC(=O)NC(COCC)C)ccncc1F.C1(=O)C(C)O1 c1(C(=O)NC(C2(O)CCN(C(=O)C(C)CO)C2)C)c[nH]c2cccnc12 c1(C(N2C3CN(C(CNC(CCC)=O)=O)CC2CC3)=O)cccc2ccccc12 C1(CC)CCCN(C(=O)Cc2cc(C)oc2C)C1C(=O)NCC(C1CCC1)OC C1(CC=C)(NC(C2CCCC2C(C)C)=O)CCN(C(=O)C(C)COC)CC1 N1(S(c2cc(Br)cc(C(=O)OC)c2)(=O)=O)Cc2ccccc2C(CO)C1 C1(F)(CNC(C2C(OCC)C2C)=O)CCCN(C(c2cc(C)cnc2C)=O)C1 N1(C(C(C(=O)N(C)C)(C)C)=O)C2CCCC1CN(C(C1(C)CCCCO1)=O)C2 CCCC(CNC(C1CN(C(C)=O)C1)=O)NC(=O)Cc1csc(S)n1 C1(C(=O)OC)CCC(O)CN1C(c1ncc(C)s1)C(=O)NCCOCC1CC1 N1(C(CNC(CCC)=O)=O)CC(N(C(=O)C=Cc2cnc(C)s2)C)C(F)C1 C1(CC)CCN(C(c2nc(Cl)cs2)=O)C1CNC(C1(NC(C)C)CC1)=O C1(C(=O)Nc2c(C(N)=O)scc2)CN(C(c2cncs2)=O)CCS1 N1(C(c2c(CNC(C3C(C)CCOC3)=O)ocn2)=O)CCC2CCCC12 CCC(CC(=O)NCC=CCNC(c1cc(CO)oc1C)=O)c1ccccc1 C(=O)(CCC(F)(F)F)NC(COC)CNC(=O)CC1CC(C)C1 C1(C)(CNC(C(CC)O)=O)COCCN(C(c2cc(C3(C)CC3)on2)=O)C1 Cc1cc(F)cc(C)c1C(N1CC2CC1CN2C(c1ncc[nH]1)=O)=O N1(C(C2(O)CC2)=O)CCCC(c2cn(Cc3ccc(OC4CCCC4)cc3)nn2)C1 CCCC(CCCNC(=O)CCc1cc(C)[nH]n1)NC(=O)Cc1ccc(CC)cc1 C=CC1(C(=O)Nc2ccc(O)cc2C)CCN(C(C2CNC(=O)O2)=O)C1 N1(C(C2C(COC)CC2)=O)CC2(CCN(C(C3(C4(O)CCOC4)CC3)=O)CC2)C1 CC1C(C)CCN1C(C1(CNC(=O)C=CCO)CC1)=O N1(C(C2CCC(n3cc(CN4CC5CC5C4)nn3)C2)=O)CC=CCC1 c1(CN)cn(CCO)c2ccccc12.C1(OC(F)F)(COC)CCOC1 CC1CN(C(=O)C=Cc2ccc(Cl)cc2)CCN1C(C1CCC(=O)N1)=O N1(C(C2(c3ccsc3)CC2)=O)CCCC1CNC(C1(C(=O)NC2CC2)CC1)=O CC(C)CCC=CC(N1CCC(CNC(c2coc(Cl)n2)=O)C1)=O c1(CC(=O)N(CCCNC(C2CC23CCC3)=O)CC)ccc(OC)c(OC)c1Cl C(=O)(C(C)=CBr)N(C(C)CN(C(=O)CCSC)C)C.CO C1(C2CCN(C(=O)Cn3ncc(Br)n3)C2)(NC(=O)CC2CCCOC2)CC1 Cc1cc(CO)ccc1C(=O)NCC1CCC(C(C)(C)C)O1 C#Cc1ccc(F)c(C(=O)NC(C)(C)CN(C)C(c2c(C)n[nH]c2C)=O)c1 C(=O)(C(C)CC(C)(C)C)NC1CCC(CNC(C2(COC)CCCC2)=O)CC1 C1(C(N(CC(C)NC(c2c(CC)non2)=O)C)=O)CC12CCOCC2 CC1(C)C=CC(N=c2[nH]c(=NCC3(C)CCCOC3)[nH]c3c2COCC3)CC1 C(=O)(CCCC(=O)NC(C)CCCCNC(=O)C(C)n1ccnc1)NC(C)C C1(CN(C(C2CC(=O)C2)=O)CC)CCCCN1C(=O)CCC1CCOC1 C1(CC(=O)NCC2CCCC2C2CC2)CC2(CC2)CN1C(=O)C1=CCCSC1 c1(C(=O)NCC(C(C)(C)C)NC(c2cc(CC)on2)=O)cc2c(Cl)nccc2o1 CC1CC(NC(=O)CNC=O)CN(C(=O)CCCc2ccnc(Br)c2)C1 C1(C(=O)NCC(c2cccnc2)C)COC2(C1)CN(C(=O)C=C1CCC1)C2 c1(OCC)ncccc1C(=O)NC1CCC(CNC(=O)C(CC2CC2)OC)C1 N1(C(C(C)OCC#C)=O)CCCCC1CNC(=O)CC1CSCCS1 C1(N(C(CCC(=C)Cl)=O)C)CCN(C(c2cccc(C(=O)OC)c2O)=O)CC1C N1(C(Cc2nnc(C)s2)=O)CC(NC(C2CCCC2(F)F)=O)C2(CC2)C1 c1(C(=O)NCC(C)N(C)C(c2ccc(S(N)(=O)=O)s2)=O)ccc2c(c1)CN(C)C2 C=CC1(C(=O)NC2(CO)CN(C(=O)Cc3csnc3C)C2)CCC1 C1(CNC(C(CC)n2cncn2)=O)CCCC2(CN(c3nc(C#N)c(Cl)s3)C2)O1 N1(C(=O)CNc2cccc(C(=O)NC3CC3)c2)CCCC2CN(C(N)=O)CCC12 c1(C(=O)NCCC2(O)CCCN(C(c3c(C)scc3)=O)C2)ccc2sncc2c1 C=CC(C)(CC)C(=O)NC1COCCC1NC(=O)CCc1ncc(C)[nH]1 N1(C(C=CCOC)=O)CC23CCCC2(C1)CN(C(=O)CC1CCC(OC)CC1)C3 C1(NC(C2(CCCC)CC2)=O)CN(C(c2[nH]c(C)cc2C)=O)CCC1C c1(C(N2C3C(N(C(c4c(C)cnn4C)=O)C)CC(C3)C2)=O)[nH]cc2c1CCCC2 C(=O)(CS(=O)CCC(F)(F)F)N1CCN(C(c2c(C)con2)=O)CC(O)C1 C1(NC(c2c(CC=C)cccc2)=O)CCN(C(c2ccco2)=O)CC12CCC2 C=CCC(C)(CC)C(=O)NCC(C(=O)NCCC(=O)OC)OC C1(C(=O)NCCOCCCN(C)C(C2CCS(=O)CC2)=O)CC(F)C(=O)N1 c1(C(N(C2CN(C(=O)C(C)(C)C(N)=O)C2)C)=O)c(N)ccc(F)c1F N1(C(CN(C2CCSC2)C)=O)CCC(CO)(CNC(=O)CCC2CC2)CC1 C1(NC(C(C)c2ccco2)=O)CN(C(=O)C=CSc2cncs2)CC1C1CC1 O=C(CC1COCc2ccccc21)NC12CC(NC(c3cc(O)cs3)=O)(C1)C2 N1(C(c2cnc(OCC)s2)=O)CCN(C(=O)C(=Cc2cccc(F)c2)F)CC1C C(CN=c1cccc(S(=O)(=O)NC2CCCC2C)[nH]1)c1nccc(C)n1 C1(NC(c2scc(C)c2Cl)=O)CC2(CCC(NC(=O)CC3CCCC3O)CC2)C1 c1(-c2c(C)occ2)nc(CCC2CCOC2)n(-c2ccccc2)n1 CC1(C)OC2(CCN(c3cc4ncnn4cn3)CC2)NC1=O n1(CCC)ccc(C(=O)NC2(CNC(=O)CCCNC(N)=O)CCC2)n1 C1(C(=O)NCC(CC)(CC)NC(=O)COc2cc(C)on2)CC1C1(C)COC1 c1(C(=O)NC2C(NC(c3ccc(C)s3)=O)C2)cc2n(n1)CCCNC2=O C12(NC(Cc3ccc(C)s3)=O)CCCC1CN(C(=O)CC1CC=CC1)C2 C1(O)(CCNC(C2CC(N(C)C)C2)=O)CCCN(C(=O)Cc2nc[nH]n2)C1 C1(CC)(NC(c2ccc([N+](=O)[O-])o2)=O)CCCN(C(=O)CNC(N)=O)C1 N1(C(C2C(C)CCOC2)=O)C(C(=O)NCC(CO)C2CCC2)CCC12CC2 C1(CC(=O)NCCN(C(C2COCCO2)=O)C2CC2)CC2(COC2)C1 CN1CCN(CCC(N2CCC(OCCNC(=O)C(C)(C)N3CCC3)C2)=O)CC1 C1(N(C(C(CCOC)C)=O)C)CCCC2CN(C(c3cncc(C)n3)=O)CC12 N1(C(C=C(CC)CC)=O)CCN(C(c2nc(CC)ncc2N)=O)C2(CC2)C1 c1(C(N2CC(CN(C(CN(CC)CC)=O)C)C2)=O)ccc(O)c(C(C)C)c1 C(=O)(C1=CCCOC1)NC(CC(=O)NC(C)(C)CCCF)CC1CC1 c1(C(=O)NCC(CNC(C(CCC#C)O)=O)OC)cc2c(C)cccn2n1 c1(C(N(C2CN(C(c3cccc(NC(C)=O)n3)=O)C2)C)=O)noc(C)c1[N+](=O)[O-] c1(SCC(=O)NCC(c2ccccc2)CNC(C(F)OC)=O)n[nH]c(O)n1 N1(C(C=C(C)C(C)C)=O)CCCC(C)(CNC(C2(N(C)C)CCCOC2)=O)C1 C(=O)(C(CC(C)(C)C)OC)N1CC(O)(C(C)NC(C2C(=C)C2)=O)C1 c1(OC)ccc(Cl)c(C(=O)NCC(C)NC(C2CC(=O)NC(=O)N2)=O)n1 C(=O)(C1=COCC1)N(CC(C)C(=O)NC1(CCOC)CC1)C C1(CNC(c2cc(CCC)n(C)n2)=O)CC2(CO1)CN(C(c1cc(Cl)cs1)=O)C2 C(C(C)CC(=O)N1CCSCC1CCNC(=O)COC1CC(F)(F)C1)OC N1(C(CCC(C)(F)F)=O)CCCC2C1CCCCN2C(C1CC=CC1)=O CCC(C#N)(CC)C(=O)NCC1CC(CNC(=O)C(C)(Cl)Cl)CO1 CCCC(CC(=O)NCCC(O)C1CCCC1)NC(c1cncnc1)=O C1(C2C(=O)N2)CCC(F)(F)CC1.C1(C(=O)OC)SCCCN1C(C)(C)C N1(C(c2c(-c3cn(C)nc3)ocn2)=O)CC2CC1C2CNC(c1cccnn1)=O CC12CCCC(C(N3CCOC(CNC(=O)CCC4CC4(F)F)C3)=O)(CO1)C2 c1(NC(C)=O)cc(Br)c(F)cc1NC(=O)C(=O)NCC1CN2CCCC1C2 C1(OC)CC(CNC(=O)Cc2csnn2)N(C(c2cn(CC(F)F)nc2C)=O)C1 CC1CCc2n[nH]cc2C1C(=O)NCc1cccc(NC(=O)NC2CC2)c1 N1(C(C(F)OC)=O)CCC2(C1)CN(C(C1CC3OC(=O)OC3C1)=O)C2 N1(C(C2C(CC)C2)=O)CCC2CN(C(C3COC(=O)O3)=O)CC2CC1 C1(C)(CNC(CC2CCC(NC(C3CC(=C)C3)=O)C2)=O)C=CCCC1 c1(C(=O)OC(C2CC(NC(=O)OC)C2)=O)cccc(CO)c1 C1(C(=O)OC)CC=CCC1C(=O)Nc1ccc(N2CCN(S(=O)(=O)CBr)CC2)cc1 c1(C(=O)OC)nc(=NCC2CCC(NC(c3cnoc3C(C)C)=O)C2)cc[nH]1 c1(OC)nc(C(=O)NC2CC(C)(NC(c3cncc(F)c3)=O)C2)sc1C n1(CC)nc(C)c(NC(C2CCC2CNC(=O)CC(C)C(F)F)=O)c1C N1(C(CCCC#CC)=O)CC(NC(c2cnc(C(F)F)s2)=O)C2(CCOCC2)C1 CC1CCC(NC(=O)CCC(C)(F)F)CN1C(=O)CC1CC2(CCC2)CCO1 C1(CNC(C2C(SC)CC2)=O)COCCN1C(c1cc(C(N)=O)co1)=O c1(C(=O)NC(C(C)C)C(=O)NCC(C)(C)NS(C)(=O)=O)cc(O)nc(O)n1 c1(C(=O)NCCC2(NC(c3cccc(C)n3)=O)CC2)nccc2ccsc12 Cc1nscc1C(=O)N(CC(C)NC(C1CC1F)=O)C Cc1cccc(C(=O)NC2CCC(C)(CNC(c3cccc(O)n3)=O)C2)c1C c1(CC)ccc2occ(C(N3CCC(N(C(C)C(C)C)C)CC3)=O)c2c1.OCC Cc1cc(C(=O)NCC2(C(=O)Nc3cc(Cl)ccc3F)CC2)cc(C)c1F C12(CNC(C=CC)=O)CC(COC)(CN1C(=O)CC1CCCCC1F)C2 N1(C(c2c(C)ncc([N+](=O)[O-])c2)=O)CCC2(CC1)CN(c1ncns1)CCO2 c1(C(N2C(C)(C(=O)Nc3sc(COC)c(C)n3)CC2)=O)ccc([N+](=O)[O-])cc1 C1(C(=O)NCC2OCC(C(=O)NC(C(=O)N(C)C)CO)C2)CCC2(CC2)C1 c1(SC(c2n(CC=C)nnn2)Cc2ccco2)cc(Cl)ccc1F C(=O)(C(C)CC(C)C)NC(c1c(CC)cccc1)CNC(=O)CC1CC1 c1(CNc2scc(-c3ccc(OC)cc3)c2)ccc(C2=CCCCC2)c(C)n1 N1(c2ccc(OC)cc2)C(=O)NC2(CCC(C)(C)CC2)C1=O Cc1ccc(CN2CCC(NC(=O)CCc3cccc(F)c3F)C2)c(F)c1 N#Cc1ccc(Br)c(C(=O)NC23CC(C(N4CC5C=CC4C5)=O)(C2)C3)c1 c1(C(N2CCC(C(C)NC(c3ccnn3C)=O)C2)=O)ccc2c(c1)CC(C)(C)O2 C[Si]1(C)CCCCN(C(C2CC(O)CN2C(c2cscn2)=O)=O)C1 c1(NC(=O)NCCc2ocnc2CO)cccc(C2(F)CC2(F)F)c1 C(C)(C)(CCC(=O)N1CCC(C)C1CNC(=O)CCCn1ccnc1)OC c1(CSC)ncc(C(C(=O)NCCCOC)N(C2CC(CC)C2)C)[nH]1 Cc1cccc2[nH]cc(CCNC(=O)CC3CCC(C#N)C3)c12 CCCCC(CNC(=O)COc1ccsc1Cl)NC(C1CCC1C(F)F)=O C(=O)(CCCCC(=O)N(C)CC1CCCC(NC(=O)Cn2nnc(=O)[nH]2)C1)OC c1(C(C)=O)ccc(C(=O)NC2CCN(C(C3CCCC3C)=O)CC2C)cc1F c1(C(=O)NC2CC3CN(C(CC(=O)NC)=O)CC32)ccc2oc(C)nc2c1 CCCC(CCCO)C(=O)NCC1CC2COCC2N1C(=O)CN(C)C(C)=O C1(NC(c2onc(OC)c2Br)=O)CN(C(=O)CCCCSC)CC12CC2 C(=O)(C1=C(C(F)F)N(C)C(=O)N(C)C1c1csc(N2CCOCC2)c1)OC C1(C)(CC(=O)NCC(C)CNC(=O)C(c2cscc2Br)=O)CC(F)(F)C1 c1(-c2nnc(N3CCC(COC)C34CCC4)n2C)ccc2c(c1)OCCO2 C1(NC(CN(CCC)C)=O)CN(c2ccnc(-c3cccc(Cl)c3)n2)CCC1C c1(C(=O)NCCCN(C(C(C(C=C)C)C)=O)C(C)C)cc(S(N)(=O)=O)ccc1C C1(C(=O)NC2CC(CCNC(c3sccc3OC(F)F)=O)C2)CC2C=CC1CC2 C1(C(=O)NCC(=O)NCC2CN(C(c3ccccc3)=O)C2)CCC2(CCC2)CC1 C1(C)(C(=O)NCc2ccc(OC)c(C(F)(F)F)c2)CCOC2(CCC2)C1 c1(NC2CCC(C(O)CN3CCCC3)C2)ncnc2ccccc12 N1(C(CC2N(CC)CCOC2)=O)CCN(C(C2CNC(=O)N2)=O)C(CCO)C1 c1(NC(C2CCC(CNc3ncncc3Br)CC2)=O)cc(F)cc(F)c1 C1(NC(C(CC)F)=O)CCC2CN(C(=O)Cc3ccc(O)cn3)CCC2C1 Cc1cccc2cc(C(N3CCC3CNC(=O)C(F)(F)C(F)(F)F)=O)[nH]c12 C(C(C(=O)N1CCSCC1CCNC(=O)C(C)CC(C)C)C(F)(F)F)OC CC(C)(C)CC(O)CC(=O)N1CCC12CN(C(=O)C(CCO)c1ccccc1)C2 C1(O)(CNC(CCCOCC)=O)CCCN(C(=O)Cc2csc(C(C)C)n2)C1 n1(CCCCC(N2C3CC(NC(CCOC)=O)C(C3)C2)=O)ncc2ccccc12 N1(C(c2nc(CCC)oc2)=O)CC2CC1(CNC(c1cc(OC)nn1C)=O)C2 C1(NC(C2N(C(N)=O)CCC2)=O)CCC2CC1CN2C(=O)C1=CCCCC1 C1(NC(c2cc(C)no2)=O)CC2CN(C(=O)COC(F)(F)C(F)(F)F)CC2C1 C1(CC(=O)NC2C(NC(c3ccn(CCF)n3)=O)CCCC2)CCCCC12CC2 N1(CCCC)CCC(NC(=O)Cn2ccc(Br)n2)C(C)C1 c1(N(C)C)ncc(C(N2CC(CCNC(=O)CSc3ccsc3)(OC)C2)=O)cn1 C1(NC(=O)C(O)C2CC2)CN(C(c2ccnc(S)c2)=O)C2(CCCCCC2)C1 c1(NC(C2OCCN(C(C3CCC(C)O3)=O)C2)=O)ccc2ncccc2c1C#N N1(CC)CCOC(CNC(=O)COC2CC(NC(c3ccc(Cl)cn3)=O)C2)C1 C1(C(=O)NCCCOC=C)CC(F)CN1C(=O)C(C)CCO C1(C(=O)NC(c2cncnc2)C(=O)NC(C=C)(C)C)CCN(C)C(=O)C1 C1(C(=O)NCCOCCC#C)CC12CC(NC(=O)C=CCCC)C2 C=C(C)C1OCCC1C(=O)NCCC1CSCCN1C(c1cncnc1C)=O C1(CNC(C2CC(C)C2)=O)C(C)CCCN1C(c1cc2n(n1)CCO2)=O c1(C(=O)NC2CC(NC(Cn3c(C)c(Cl)cn3)=O)C2)cccc2c1OCCN2C C(=O)(CCS(=O)(=O)C1CCCC1)NCCC1(NC(CC2C(C)(C)C(O)C2)=O)CC1 N1(C(Cc2cccc(OC)c2Cl)=O)CCCC(C2CN(C(=O)CC(C)SC)C2)C1 C(CCN=C(NC1CCC(=O)N1)N1CCC(C2CC2)C1)OCC N1(C(CN(C2CC2)CC)=O)CCCc2c(NC(C)=O)cccc21 N1(CC(=O)N(C)Cc2ncc(F)cn2)CCCC(N(C)C)CC1 c1(C(=O)NC2C(C)CN(C(C3C(C#N)C3(C)C)=O)CC2)ccn2c(O)nnc2c1 C(=O)(C(C1=NOC2C3CCC(C3)C12)N1CC(F)(F)CC1(C)CO)NCC(=C)C N1(C(CC=CCCCCC)=O)CC(C(=O)NCCc2cnc(C)cn2)C(C)(C)C1 n1(CC(N2CC(CNC(C3CCC(C)(CC)O3)=O)(CO)C2)=O)ncc(C)cc1=O C(N=c1cccc(S(=O)(=O)N2CCCC2C2CCOC2)[nH]1)C1(C2C(F)(F)C2)CC1 C(C(N=[N+]=[N-])C(=O)N1CC(CNC(=O)CC2CSCCS2)(COC)C1)OCC C1(N(C)C(C2C3CCCC23)=O)CN(C(C2(CCc3ccccc3)CC2)=O)CC1F C1(C(N(C)Cc2ccsc2)=O)CCCN1C(c1cc(Cl)cs1)=O C(=O)(C(C)C(C)S(C)(=O)=O)NC1CCN(C(c2ccc(C(C)C)c(Cl)c2)=O)CC1C Cc1c(Br)ccc(F)c1C(=O)NC(C)CCNC(c1cnc2n1CCC2)=O Cc1cnc(CNCC2CC(C(F)(F)F)CO2)s1 N#Cc1ccc(F)c(Cc2cn(C3CN(C(c4cnc(C#N)s4)=O)C3)nn2)c1 c1(N2CCc3n(NCC)cnc3C2)nc2c(c(=NC3CCC(CC)CC3)[nH]1)SCC2 C(=O)(C(C)(C)CCSC)N1CC2C(NC(CCOCC(C)C)=O)(C2)C1 C1(CNC2C(Cc3c(C)oc(-c4ccc(Cl)cc4)n3)C2)CCC2(CC1)CC(O)C2 c1(NC(C2CC(NC(C=CCN(CC)CC)=O)C2)=O)cc(C2CC2)nc(Cl)c1 c1(CNC(C2N(S(CC)(=O)=O)CC(C)C2)=O)cc(Cl)c(F)cc1F N1(C(C=C(CC)CC)=O)CC2CCCC2(CNC(c2ccc(C#N)c(C)n2)=O)C1 CCC(CC(C)C)C(=O)NCC1CCC(CNC(C23CCC2C3)=O)CC1 C=CC1(C(=O)NC2CC(C(N)=O)(SC)C2)CCN(C(=O)CC2CCCCCC2)C1 C(CO)(CCCCNC(=O)CCCC(C)O)NC(C1CC(C)OCC1)=O c1(C(C(=O)NC2C(NC(c3n(CCC)ccc3)=O)C2)C2CC2)ccc(F)cc1 N1(C(c2c(C)occ2)=O)CCC(CNC(C2(C3CCCO3)CCC2)=O)CC1C c1(C(=O)NC(C(C)C)CCNC(=O)CC(C)c2ccco2)ccn(C)c(=O)c1 C(C)(C(C)(C)C(=O)NCC1(C2CC2)CCCO1)NC(C(=O)NCC)=O c1(C(N(C(C)CNC(c2cc(-c3ccns3)on2)=O)CC)=O)cc(C)cs1 C1(CNC(CC(CCC)O)=O)CC2COCC2N1C(C1CCCC(O)C1)=O CC(C)(C)C(C#N)C(=O)N1Cc2[nH]nc(C(=O)NC3CC4(CCCCO4)C3)c2C1 CCCCC(CNC(=O)COCC)NC(c1nc(C(C)=O)sc1C)=O C(=O)(CCC(F)(F)F)N1CC(C(C)NC(=O)CC2(C)CCCO2)OCC1 c1(C(N2C(CN(C(=O)CC3CCCO3)C)CCCC2)=O)cccn2cncc12 c1(COC)cnc(O)c(C(=O)NCCOCCNC(=O)CSCc2nccn2C)c1 c1(N(C)C)ccc(NC(=O)NCC2(C(F)(F)F)NC(=O)NC2=O)cn1 c1(C(=O)NC(c2cccnn2)=O)occc1CNC(C1CC1CCOCCO)=O c1(OC)cc(CCC(N2CC3CC2CN3Cc2cc(Cl)cnc2Cl)=O)ccc1O c1(CCC(=O)NC2(C)CC(NC(Cc3c(C)noc3Cl)=O)C2)cc(F)ccc1F C1(C(N2CC(C(C(=O)NCCCc3cccs3)OC)C2)=O)(SC)CCC1 CC1CC(NC(=O)Cc2ccc(Cl)cn2)CN1C(c1ccccc1CN(C)C)=O C1(C(=O)NC(C)CCN(C(=O)C(O)CC2CC2)C)CCC(C)CC1 C1(C)(C(N2CC(C(C)NC(C3CCOC3)=O)C2)=O)C=CCC1 CCC(C)CC(C)NC(C1(NC(C2CC(C(=O)OC)C2)=O)CC(F)(F)C1)=O c1cc2n(c1)CCCC2.C(CP(C)(C)=O)(C(N)=O)c1sccn1.C12(CCCN1)C1=CC=C2OC1 C1(NC(Cn2c(C(C)C)nnn2)=O)CN(C(=O)COCC(F)F)C2CC12 c1(C(N(C2CCN(C(=O)CC3(CC)CCC3)CC2)CCC)=O)cnc2sccn12 c1(-c2c(SC)cccc2)ccc2c(CNC(c3cc(F)ncc3F)=O)n[nH]c2c1 C(=O)(C(O)C(C)CC)NCc1c(C(=O)NC(C#C)C(C)OC)cccn1 N1(C(CC2(COCC)CC2)=O)CCC(C)C1C(=O)Nc1cccc(C(=O)OC)c1.OCC c1(CC(N2CC(O)(CCNC(C3CC3F)=O)C2)=O)c(O)ncnc1O c1(OCC)ccc(N(C2CCNC2)C)cc1 CCCC(F)C(=O)NCC(CC(=O)NC(C)(CC)CO)C1CCC1 C(=O)(CC(O)CNC(c1c(C)noc1C)=O)NC(c1ccn(C)n1)CC c1(-n2c(C)nc(C(=O)NCCC(Cl)Cl)n2)ccc(Cl)cc1Cl C#CC1(NC(=O)C(O)CNC(c2cc(C)nn2C)=O)CC2CCCC12 N1(C(c2ccc(OC)cc2N)=O)CCC2CN(C(C3(CF)CC3)=O)CC12 CC(CC1CCC1)C(=O)NC1CC(CNC(c2c[nH]nc2C(C)(C)C)=O)C1 C1(CC=C)(NC(=O)C(C2CCN(C(c3ccc(Cl)o3)=O)C2)C)CC=CCC1 N1(C(C)=O)CCC(C(=O)NC2(C3CN(C(c4sccc4C)=O)C3)CC2)C(O)C1 N(C1CCc2cccc3cccc1c23)C(N1C(CCC=C)CCC1)=O C1(N(C(=O)Cc2cc(-c3ccco3)on2)C)CCC(NC(C2(C#N)CC2)=O)CC1 c1(C(=O)NCC(CCOC)NC(CC(C=C)C)=O)cccc2occc12 c1(C(CC)C(=O)NCC(O)CNC(=O)Cc2cnn(CC)c2)c(C)noc1C C(CCN=c1[nH]nc(C(C)(C)C)s1)N(C(C1CCCN(C)C1)=O)CCO C1(CC(N2CC(OCCC(=O)NCCSCCC)C2)=O)CCCC1C S(=O)(=O)(CCCS(=O)(=O)Nc1ccc(CN2CCCC2=O)cc1)N(C)C C1(NC(c2c(C)scn2)=O)CN(C(c2cc3c(o2)CCCC3)=O)C2CCCCC12 C1(NC(CN(c2ccccc2)CC)=O)CCCC(CNC(=O)CC2CC(F)C2)C1 c1(CNC(CNC(CNC(c2c(C)[nH]cc2)=O)=O)=O)ncc(Cl)cn1 C1(OC)CC(CNC(c2cc(CCO)on2)=O)N(C(=O)CC2C(=O)NN=C2C)C1 C1(CC)CN(C(=O)C(=O)NC(C)C)CCN1CCCn1cncn1 N1(C(C2(S(C)(=O)=O)CC2)=O)CC(NC(c2nncs2)=O)C2(CCOCC2)C1 N1(C(CC(C)CNC(=O)OC(C)(C)C)=O)CCCC(O)(NCNC(=O)C(C)(F)F)C1 c1(C(=O)OC)ccc(C(=O)NCC(CO)NC(C2CCC2)=O)c(Cl)c1 c1(C(=O)NC2CCN(C(c3cc(OCC)n[nH]3)=O)C2C)cnn2ccc(O)nc12 C1(NC(=O)COC2CCOC2)CC2CCC(C1)N2C(c1csc2cncn12)=O Cc1cc(C)c(C(N2CCCC(NC(=O)C3=CSCS3)C2)=O)cn1 C(C(C)(C)C(=O)N1CCC(C(C)C)C1)N(C(C(CC)=CCCC)=O)C c1(NC(=O)C(C)Oc2ccccc2)ccn(C)n1.C1(=O)CCN1CC CC1NC(=O)CCC1CNC(=O)CN(C(c1ccc(Cl)o1)=O)C1CC1 Cc1cc(O)ccc1CNC(=O)C(Cc1cn[nH]c1)NC(=O)CC(C)C(C)C c1(OC)cn(C2CN(C(c3ccc(C(C)=O)[nH]3)=O)C2)nn1 N1(C(C(CC=C)CC(C)C)=O)CC2(CCN(C(=O)CCSC)CC2)C2COCC12 C(CCC(C)(C)NC(=O)C(CC)NC(C)=O)NC(C(C)OCCCC)=O C1(CNC(C2CC(CCC)C2)=O)C2CN(C(C3(C)CCCOC3)=O)CC12 c1(NC(CCC2(NC(C(CC)OC)=O)CCCC2)=O)cccc(OC)c1 c1(C(=O)NCCN(C(C2C(OC)C2)=O)C)ccc(C#N)cc1 c1(CC(=O)NCCC2(CNC(C(CCC)OC)=O)CC2)ccc2c(c1)NC(=O)C2 C1(CNC(c2nnc(O)nc2O)=O)CN(C(=O)C(N2CCCC2)C2CC2)CC1(F)F C1(C(=O)NCC2OCCCN(C(CCC)=O)C2)CCN2CCCC2C1 C1(C(=O)NC2CC(C(F)F)(NC(CC3(C=C)CCC3)=O)C2)CC12CCCC2 c1(C(=O)NCC2(C(=O)NCCCC(O)CO)CC(=C)C2)cc(C)c(C)o1 N1(C(C=C(CC)CC)=O)CCC2(CCCN2C(c2ccc(O)c(N)n2)=O)C1 C1(OC)CN(C(c2sccc2C#N)=O)CCC1NC(=O)C(F)C(C)(F)F C1(C(=O)OC)CN(CCOCCNC2(CC(C)C)CCC2)CC2(CCC2)O1 C#Cc1cnn(C)c1C(=O)NCC1CN(C(=O)CC2CC(F)(F)C2)CC1(C)C c1(C(N2CCC(N(C(CNC(CC)=O)=O)C)C2)=O)cc(S(N)(=O)=O)co1 c1(C(N2CC3C(CNc4c(C#N)cccn4)C3C2)=O)ccnc2[nH]ncc12 N1(C(c2ccc(CC)o2)=O)CC(NC(c2ccc(C#N)s2)=O)C(C)C1 N1(CC(=O)NCC(C)(C)CO)CC2CCC(C1)C2N.C12CCN(CC1)C2=O C=CC1(NC(=O)CC(C)C)CCN(C(=O)C(C)(C)C(C)O)CC1 CCC(CC(=O)N1CCOC(C(=O)NCC2(O)CC(CF)C2)C1)SC C1(NC(c2ccc(C)c(C)c2)=O)COC2CN(C(C3CC4(CCC4O)C3)=O)CC12 C(C)(C)(C(=O)NCc1cn(CC(=O)NCC2CCN(C)C2)nn1)OC C1(CNC(CCc2ccn(C)n2)=O)(NC(C2(C(F)(F)F)CCO2)=O)CCCCC1 N1(C(c2cnc(CC)s2)=O)CCCC2(NC(=O)C=Cc3cc(C)no3)CCCC12 C(=O)(CC(CNC(=O)CCCC1N=N1)C1CCC1)NC(C)Cn1cccn1 c1(N(C(C(=O)NCCCF)C2C(CC)C2)C)ccccn1 N1(C(CCCCOCCC=C)=O)CCCN(C(=O)CC(C)(C)C(=O)OC)CC1C N1(C(CCN(CCC)C)=O)CCc2ccccc2C1CNC(c1cc(C)[nH]n1)=O c1(C(N2C3CCC(CNC(COCCC)=O)(C3)C2)=O)cc(C)c2c(c1)CCC2 N1(C(C(C)C2CC2)=O)CCC(C2CCN(C(=O)CNS(=O)(=O)N(C)C)C2)CC1 c1(OC)cc(C)ccc1OCC(=O)N(CC(O)CNC(=O)Cc1csnn1)C C1(C(N2CCN(C(CCSCC)=O)C(COC)C2)=O)CCc2cnnn2C1 Cc1[nH]c2ccc(F)cc2c1CC(=O)NCCN(C)C(C1(F)CCCOC1)=O c1(C(=O)NCC(CNC(C2CC(CN(C)C)C2)=O)O)cc(F)c(F)cc1Cl C1(CNC(=O)COC2CCN(C(c3cccnc3)=O)C2)CCC=CCC1 C1(C(=O)NC2CCC(C(=O)NCCC3CCOCC3)C2)CCC(C2CC2)C1 c1(CC)ccc(C(=O)NCC2COCCN2C(c2csc(Cl)c2)=O)cc1[N+](=O)[O-] N1(C(CCc2ccc(OC)cc2)=O)CCC2CCCN(C)C2C1 C(=O)(CC(C(F)(F)F)NC(C1CC2(CCO1)CC2)=O)NCC(C)(O)CO C1(CC#C)(C(=O)NCCCC2CN(C(=O)CC3CCOC3)CCO2)CCCCO1 c1(C(=O)NC(c2cccc(Cl)c2)CNC(C(CC)C#N)=O)c(OC)cccc1F C1(NC(CSCc2cccc(C)c2)=O)CCN(C(=O)C=CC2CCC2)CC1C c1(CC(=O)NCC(CC=C)NC(C2CC3C=CC2C3)=O)ccc(Cl)nc1 n1(C(C)C)ncc(F)c1C(=O)NC1CC(C)N(C(=O)CCN2CCCCC2=O)C1 C1(C(N(CCOCC)C)=O)CN(C(C2(C)CCCS2)=O)CC12CC2 C(=O)(CCS(C)(=O)=O)NCCCNC(C1(CC2CN(C)C(=O)C2)CCSCC1)=O CC1(CNC(=O)CCNC(c2ccon2)=O)CCCC1O N1(C(C2=CCC(NC(C3(CC#C)CCCO3)=O)C2)=O)CC(C)(C)OC(C)(C)C1 c1(C(=O)NC2C(C)N(c3cnc(F)cn3)CC2)coc2c1NC(=O)CCC2 CCCC(C(=O)OC(C)(C)C)C(C)C.C12(C)CCCCN1C(=O)N2 c1(C(CNC(c2c(C(C)C)cco2)=O)NC(=O)CC(C)(C)C)ccc(F)cc1F C(=O)(C1=C(C)CC1)NCC1(CO)CN(C(C(C)(c2ccccc2)NC(C)=O)=O)C1 N1(C(C(C)OCC=C)=O)CCC2CN(C(=O)C=Cc3cc[nH]c3)CC2C1 N1(C(CC2CCCC(CNC(=O)OC(C)(C)C)C2)=O)Cc2cc(O)nnc2C1 C(=O)(C1=C(C(=O)N2CCCC2(C(=O)OC)C(C)C)CC1)OC C1(N(C(=O)C=Cc2ccoc2)C)CN(C(c2ccoc2Cl)=O)CC1(C)C c1(C(=O)NCc2c(C(N3CC(CO)CC(C)C3)=O)occ2)cc2ccccn2c1 N(C(=NCC1CC1)N1CC(c2ccccc2)C2(CCC2)C1)C(COC)C Cn1ncc2ncc(C(=O)NCC=CCNC(=O)Cc3ccncc3Cl)cc12 c1(C(=O)NC(CNC(c2cc(OCC)cc(=O)o2)=O)C)cc(C)cc(OC)c1O C1(CC(=O)NCCOC2CC(CF)C2)CC(C2CC2)C1.C1(C2(O)CCC2)C(=O)N1 C1(C(N2CC(CC(=O)Nc3cnnc(Cl)c3)OCC2)=O)CCc2ccccc2C1 N1(C(c2c(N(C3CC3)CC)nc(C)cc2)=O)CC2CC3CC2C1C3 C(=O)(CC(C(F)F)NC(=O)C=C(C)c1ccco1)NC(COC(C)=O)CO C1(C(=O)NCC2(F)CN(C(C3CCC(C)(O)CC3)=O)C2)CCC2(C1)CC2(F)F C1(NC(CN(C2CCSC2)C)=O)CC2CN(C(c3nnc(S)n3C)=O)CC2C1 C1(C(=O)NCC2(C)C(NC(CCC3N(C)CCC3)=O)CCC2)CC2OC1C1CC21 C(=O)(CCCC(C)C)N(CCCNC(C(Br)=C(C)C)=O)CCO N1(C(CCS(N)(=O)=O)=O)CC2CC(C(=O)NOCCC(F)F)C(C2)C1 c1(C(N2CC3C(NC(c4c[nH]nc4Cl)=O)C3C2)=O)cnc2[nH]ncc2c1 C=CC1CC1(c1cccnn1)NC(C1(CSC)CC1)=O Cc1ccc(Br)cc1-n1nc(-c2ccc(Br)cc2)nc1CC(C)C1CC1 C1(C(=O)NCc2c(C(=O)NC(c3nnnn3C)C)cccn2)CCCC1C1CC1 c1(C(=O)NC2CCN(C(C3CC(=O)NC(=O)N3)=O)CC2F)cncc2sccc12 c1(SC)cccc(C(=O)NC2(C)CN(C(C34CC3C4)=O)C2)c1 C=CC1(O)CCN(C(=O)C(CC(F)F)NC(c2coc(OCC)n2)=O)C1 C12(C(=O)NC3CCN(C(CN4CC(C)C4)=O)C3)CCCCC(=O)N1CCC2 Cc1nn(CC(=O)NCc2nncn2C)c(=O)o1 C12(CNC(c3c(C(C)C)occ3)=O)CCC(C1)N(C(=O)COC1CC=CC1)C2 CC1CC(C)(NC(=O)COc2ccon2)CC(C)O1.N12CC3(CC(CO3)C1=O)C2 c1(CC(=O)NC2C(NC(C(CC)(CC)CC)=O)C2)c[nH]c2cccc(F)c12 C(CCCC(=O)NOC1CCCN(CC)C1)N(C(C(CC)CC)=O)C CCCCCC(CCCCC)C(=O)N1CC2CN(C(=O)C(C)S(C)(=O)=O)CC2C1 C(=O)(CCS(=O)(=O)N1CCCC1)N1CC(NC(COCCOCC)=O)C1.C(C)(C)C c1(C(=O)NCC(C)NC(c2noc(C)c2[N+](=O)[O-])=O)ccc2cccc(C)c2n1 C1(=CCCNC(C2(NC(C3C(CC)CC3)=O)CC2)=O)CCC(C)CC1 CCC(CCCC(=O)N1CCC(CN(C)C)CC1)NC(c1cccc(=O)o1)=O c1(CC(N2CC(F)(CNC(c3c(C)c(Br)cs3)=O)C2)=O)c(C)ncnc1C c1(CC(C(=O)NCC(C=C)O)NC(=O)C(C)SCC)cnn(C)c1O CC1CC(N=c2nc(N3CC4CCC3C4)c3cccc(F)c3[nH]2)CC(C)S1(=O)=O N1(C(c2c(CC)nn[nH]2)=O)CC(O)CC1C(=O)NCCc1nccs1 c1(CC)cc(C(N2CCCC(NC(c3ncc(F)cc3C)=O)C2C)=O)cc(F)c1 N1(C(c2ccc(C)c(O)c2)=O)CCC2(CCCC2NC(c2coc(CO)c2)=O)C1 C1(NC(Cc2c(C)n[nH]c2C)=O)CCN(C(c2cccc(O)n2)=O)CC1O C(=O)(C(C)(C(C)C)OC)NC1CCC1.CCCCC(=O)NC1C2CN(C)CC12 C1(C(=O)NCCCCCN(C(CN(C2CC2)CC)=O)C)CC(C)CC(C)(C)C1 c1(NC(C2CCC(CC)C2)=O)ncc(C)cc1S(=O)(=O)N.c1(C)cc(Cl)ccc1F CC1(F)CN(C(C2(C3CC3)CC2)=O)CCN(c2cc(O)nc(=O)n2C2CC2)C1 C1(CNC(C2N(CC)CC2)=O)(CO)CCCN(C(=O)C=Cc2ccc(SC)s2)C1 c1(C(=O)NC(C(=O)NCCC2ON=C(C)C2)(C)C)ncnc(O)c1F CC(C)(C(=O)NC1CN(C(=O)CCNC(N)=O)CC1O)C(N)=O c1(NC(C2CCCC(CC)N2)=O)coc2c(F)cc(Cl)cc12 c1(OCC(=O)NCC(C)CN(C)C(c2cc(F)c[nH]2)=O)ccc(Cl)c(F)c1 c1(C(CC(=O)N2C(CNC(c3cn(CCC)nc3)=O)CC2)O)ccc(F)cc1 N1(C(CCc2c(C)cccc2)=O)CCCC(COC)(NC(=O)C(C)P(C)(C)=O)C1 c1(C(N2CC(OCC)(CNC(=O)Cc3csc(CC)n3)C2)=O)cc(O)nnc1O CC(C)(C)CC(C(=O)NC1CN(C(=O)C2CC2)C1)N1CCCC(C)(CO)C1 C1(NC(C=Cc2ccc(SC)s2)=O)CCCCCC1NC(=O)CS(=O)(=O)N(C)C c1(C(N(C(C)CN(C(=O)C(=O)N(C)C)C)C)=O)ccc2cnsc2c1 N1(C(CC2ON=C(C)C2)=O)CCC(NC(=O)CC(=O)OCCC(C)C)CC1C c1(C(C)(C)C)ccsc1C(=O)NC1CC1CNC(=O)C(C1CC(F)(F)C1)O c1(CNC(Cc2c(C)ccs2)=O)ccccc1CNC(=O)CCC(C)C C1(C(=O)NC2CC(CCNC(CCCC=C)=O)C2)CN=C2N=CNN2C1 Cc1ccc(F)cc1-c1nnc(N2CCCN(C3CCCC3)CC2)n1CCC#N c1(C(N(CC(=O)N(CCNC(C)=O)C)CC(C)C)=O)ccc2cncn2c1 N1(C(C23C(C)OC(C)(C2)C3)=O)CC(CO)C2(C1)CN(C(c1ncc[nH]c1=O)=O)C2 C(=O)(CP(=O)(C(C)C)C(C)C)NCCOC1CCN(C(CC(C=C)C)=O)C1 N1(C(CSCC=C)=O)C2CCC1CN(C(=O)CSCCC#N)C2 C1(CNC(=O)Cn2nnnc2-c2ccsc2)CCCCN1C(C1CC(CF)C1)=O C=CCCC(=O)NC(C)C(C)NC(=O)CCNC(c1ccoc1)=O C(C)(CCCC(=O)NC(c1cnsc1)C)NC(c1c(CCC)nco1)=O C(C1C(C(=O)NC2CCN(C(C3COC(=O)N3)=O)C2C)C1(C)C)=C(C)C C(=O)(C1=C(Cl)CCC(C)C1)N1CC(CNC(c2c(C)cc(C#N)cn2)=O)C(C)C1 CC1(O)CCN(C(C2C3CCC(C3)N2C(C2(C#N)CC=CC2)=O)=O)CC1 C1(C)(CC)C(=O)NCCN1C(C1CCC2(CN(CCC(=O)NC)C2)O1)=O c1(CNC2(c3n(C(C)(C)C)nnn3)CCOC2)cc(Cl)ccn1 c1(CNC(C2CN(Cc3ccc(O)nc3)CCC2(F)F)=O)ccnc2[nH]ccc12 C1(CC(N2CCC(C)(NC(C)=O)C2)=O)CCN(CC=Cc2ccccc2)C1(C)C C1(C(N(C(CNC(c2nc(OCC)oc2)=O)C)C)=O)CC2C=CC1C2 Cc1nsc(C)c1C(=O)NCC1CC(C(=O)NCCCCN(C)C)C1 c1(CC)cc(NC(=O)C(CC)=CC(=O)N(CC)CC)no1 CC1CN(C(c2ccc(F)o2)=O)CCN1C(=O)CCCn1cncn1 c1(SC)cccc(Cl)c1.CCCC1CNC(=O)C2(CC2)C(=O)N1 C=CC(C)(CC)C(=O)N1CC(O)(C(C)NC(=O)CCC2CC(C)(C)CO2)C1 N1(C(C2C3CN(C)CC32)=O)CCCC2CN(C(c3cc(N)c(F)cc3F)=O)CC12 c1(C(N2CC(C(N3CCCCC(O)C3)=O)C(O)CC2)=O)ccc2c(c1)C(=O)NC2 S(=O)(=O)(c1ccc(C)cc1)C(CC)NC(=O)CCCc1csc2ccccc12 C1(C(N2C3(CC(C(N)=O)C3)CC2)=O)N(C(=O)C(F)C2CCC2)CC12CCCC2 c1(C(=O)NC2(C)CC(NC(=O)CCc3cn[nH]c3)C2)ccc(S(N)(=O)=O)c(Cl)c1 N1(C(C(CCC)O)=O)CCC2C(CCN2C(=O)C=Cc2ccccc2Cl)C1 C1(C(N(C(CCNC(CSCCCC)=O)=O)C)C)CCCCO1 ClC1(Cl)CC(OCCN2CCCC2c2ccncc2)C1 c1(C(N(CC(C)NC(C(C)OCCOCC)=O)C)=O)csc(Br)c1C c1(C(=O)NC(CCOC)CNC(c2cn(CCO)nn2)=O)cccc2nn[nH]c12 CN=C(NCc1cccs1)N1CCC(NC(=O)CC2CCSC2)C1 N1(C(c2cn(CC)nn2)=O)CC(NC(C2(C(F)(F)F)CC2)=O)CC12CCCC2 c1(C(=O)NC2CC(CNC(c3ccccc3)=O)C2)cc(O)ccc1O C1(CC=C)(C(=O)NC2CC(CF)C2)CCN(C(=O)CCOCC2CC2)C1 C(c1ccc(O)cc1)=C(C(N1CCC(CC=C)(NC(C2CNC(=O)C2)=O)C1)=O)C#N C#Cc1cccc(C(=O)Nc2cc(C)c(C(F)(F)F)cn2)c1.C12CC1CNC2=O CN1CC=C(C)CC1.C(=O)(C(C)(C)C(=O)N(C)CP(C)(C)=O)N1CCCCC1 C=C(C)CCCC(=O)NCC1CCN1Cc1cn(-c2ccc(Cl)c(F)c2)nn1 CCC(C)CC(=O)NCCC1CCN(C(c2ccc(-c3cnco3)cc2)=O)C1 C1(C(=O)NC2C(C)CCN(C(c3occ4c3CCC4)=O)C2)CC2C=CC1C21CC1 Cc1ccc(C2C(C)CN2C(=O)CCCN(C(C)CCO)C)cc1 N1(C(CC(CCC)O)=O)CCCCC2(CCN(C(=O)Cc3cc(C)on3)C2)C1 c1(C(=O)NC(C)C2CC2)cc(-n2cc(C3CC3C(=O)O)nn2)ncn1 CCCC(C(=O)OC)C(=O)N1CC2CCC1CC2NC(=O)C(CC)(CO)OC C1(NC(c2cnc(C)nc2)=O)CN(C(c2ccc(C(F)F)o2)=O)C2CCCC12 c1(C(N2CCC(NC(c3nncs3)C)C(C)C2)=O)ccc2cccnn12 C1(NC(C(C)(C)C2CC2)=O)CCCCC1Nc1ncc(OCC(F)(F)F)cn1 c1(C(=O)NC2CCCN(C(=O)Cn3cncn3)C2)ccc2c(c1)NCCNC2=O C(=O)(C#CC1CCCO1)NCC1(CNC(c2c(CC)[nH]cc2)=O)CC1 Cc1ccc2c(=O)c(C(=O)NC3CCC(N(C)C)CC3)c[nH]c2c1C c1(CNC(N(CCOC)C(c2n[nH]c(C)n2)C)=O)ccc(Cl)nc1 c1(C(=O)NC2C3CN(C(c4cnc(C(C)OCC)s4)=O)CC32)ccc(O)nc1Cl Cc1ccc(C(N2CC(C(C)NC(c3ncc(Cl)cc3F)=O)C2)=O)cc1[N+](=O)[O-] C#CCC(O)C(=O)N1CC2CC1C2C(=O)NC(c1cn(C)nn1)C C(=O)(CC(C)(C)C(=O)NC1COCC1NC(=O)C(C)(C)C)OC.C(=O)(CCCCO)NC Cc1ccc(C2CCCN2S(=O)(=O)CCNCC2(O)CCOCC2)cc1 C1(CNC(C(N2C(=O)CCC2=O)C)=O)(CNC(c2nsnc2O)=O)CC12CCC2 CS(=O)(=O)c1ccc(C(N2CC3=C(C2)CN(C(C2CCNC(=O)C2)=O)C3)=O)s1 N1(C(C2N(CC)CC2)=O)CCC(NC(c2cc3c([nH]2)CCCC3)=O)CC(O)C1 C1(C)(CNC(C2OCCC(C)(C)C2)=O)CN(C(=O)Cc2ccoc2)C(C)(C)C1 C1(NCc2ccn(C(C)C)n2)C(C)CCCN1C(=O)Oc1ccccc1F c1(NC(CC)Cc2ccccc2)cc(NCCCN(C2CC2(F)F)C)nc(C)n1 C12(C(C(=O)N3CC(C(=O)OC)C3)OC)CC(CO)(C1)C2 C1(NC(CSCCOC)=O)C2CC3CN(C(c4ccc(Br)o4)=O)C1C3C2 CC1(C(=O)NCCCCCCO)CCCN(Cc2ccc(Br)s2)C1 O=S(=O)(c1ccc(NCC2CCOC2)cc1Cl)NCC(F)C1CCC1 C1(CN2CC(C3CN(C(C(C)CS(C)(=O)=O)=O)C3)OCC2)CCc2ccccc2O1 Cc1ccc(C(C)C)cc1C(=O)NCC1CC(F)(F)CN1C(=O)Cn1cnnn1 Cc1csc(=NCC(=O)NCC2CC(NC(c3cc4cc(F)ccc4o3)=O)C2)[nH]1 N1(C(C2(COC)CC=CC2)=O)CCCC(NC(=O)CC2CS(=O)(=O)C2)C(F)C1 C1(C(N(C(CC)CN2CCCC2)C)=O)C(O)CCN1C(=O)CNc1ccccc1 C(=O)(C(O)C(C)(C)C)NC(CCCNC(CN1CCC(OC)C1)=O)(C)C c1(C(N2C(CNC(CC3CC(=O)NCC3)=O)CC2)=O)ccc2c(c1)NCC2 c1(CC2(N(N3CCOC(C(F)(F)F)C3)C)CC2)cccc(S(N)(=O)=O)c1 CC1(C)CN(C(=O)NCCCn2cc(C(F)(F)F)cn2)CC(c2ccccc2)O1 Cc1cc(-c2nc(-c3ccccc3)nn2C(C)C(C)C)cc(C)c1 C1(C)(OC)CCC(NC(c2csc(C(=O)Sc3ccc(C#N)cc3)n2)=O)CC1 N1(C(c2occ(C)c2)=O)Cc2occ(C(=O)NC3CC4CC(OC)C4C3)c2C1 C1(C(N(C2CC(C(=O)NCC3CC(=C)C3)C2)C)=O)COCCN1C C(=O)(C(C)CC(C)(C)C)N1CCC(NC(CCc2ccc(OC)cc2)=O)C1 C1(NC(CCCC#C)=O)(CNC(c2ccc[nH]2)=O)CCC(F)(F)CC1 C1(C(=O)NC2C(C(=O)OC)CC2)(OC)CC(CO)C1 N1(C(c2c(C)cns2)=O)CCC(CO)(NC(C2OC(C)CC2C)=O)CC1 C(=O)(NNc1ccc(Cl)cc1Cl)Nc1c(C)n(C)nc1C(F)F C(CCCCCC(=O)NCC(C1CC1)NC(C1(S(N)(=O)=O)CCCC1)=O)SC c1(C(COC(C(C)(C)N2CCCC2=O)=O)=O)cc2cscc2s1 C1(CNC(=O)CN)CCC(CNC(N)=O)CC1.N1(C(CCOCC#C)=O)CCOCC1 C1(CC)(CC)CCCN(C(c2sccc2CNC(c2cc(O)nc(C)n2)=O)=O)C1 CC(C(=O)N(CCNC(=O)CC1CSC1)C1CC1)C1=CCCC1 c1(OC)ccc2c(c1)C(C(=O)NC1CC(C)(C)C13CCC3)CCC2 N1(C(=O)Cc2nc[nH]n2)CCN(C2CN(C(=O)COCCC3CCC3)C2)CC1 c1(C(=O)Nc2ccc(NC(C)=O)c(F)c2)cc(C#N)c2cc[nH]c2c1 Cc1c(F)ccc(C(N2CCN(C(c3cn4c(n3)CCC4)=O)C3CC23)=O)c1F N1(C(C(C)SCCCC)=O)CCN(C)CC1CNC(C1CC=CC1)=O C1(NC(=O)CCc2cnc[nH]2)CCCCN(C(c2ncc(Cl)cn2)=O)C1 C1(NC(CCN(CC#C)C(C2CC2C(F)F)=O)=O)CCN(C)C(=O)C1 c1(SC)cc(C(N2CCSCC(CO)C2)C(=O)NC2COC2)ccc1OC C1(NC(Cc2c(C)cccc2)=O)CCCN(C(=O)COC2CCCOC2)C1C c1(C(N2CCCC(CNC(C3(C)CCCOC3)=O)CC2)=O)nccc2[nH]ccc12 C1(CC(=O)NCC2CCC2(F)F)C2CN(C(=O)CCn3ccnn3)CC12 C1(N(C(=O)C(O)CC2CCCCC2)C)CCCN(C(c2cccs2)=O)C1 c1(C(C)C)cc(C(=O)NC(C2CN(C(=O)CSC(F)F)C2)C)n(C)n1 c1(CNC2CCN(c3cc(C)nn3C)CC2)ccc2c(c1)CCS2(=O)=O N1(C(C2CC(F)(F)C2)=O)CCCC2(CCCN2C(=O)CSCC2CCCO2)C1 c1(CC)ccc(C(=O)NCCC2CCCCN2C(=O)CC2CCC(=O)NC2)cc1 C12(CC)COC(C(=O)N(CCCNC(=O)C(C3CC(C)(C)C3)OC)C3CC3)(C1)C2 C1(NC(Cn2ncc(C#N)c2)=O)CC(NC(c2cscc2Cl)=O)C12CCC2 C1(NC(c2c(COC)cccc2)=O)CC2CCC(C1)N2C(=O)CSC(F)(F)F C(CCC(C(=O)Nc1cc(C)cnc1OC)NC(=O)C=CC1CCOC1)OC N1(C(C(C)OCC(F)(F)F)=O)CCC(CCN(C(=O)C(C)c2cccs2)C)CC1 C=CCCCC(C(=O)NC1CCC1)NC(c1ncncc1F)=O N#Cc1nc[nH]c1C(N1CC2C(CNC(c3ncc[nH]3)=O)C2C1)=O C12(CNC(=O)CSc3n[nH]c(O)n3)CCCCC1CN(C(=O)Cn1cnnn1)C2 C1(C(C)(C)C)(CNC(=O)CC2C=CCC2)CCN(C(c2ncc(F)cn2)=O)C1 c1(C2OCCN(C(c3cccc(OC4CCOC4)c3)=O)C2)cc(F)cc(F)c1 N1(C(CSC)=O)CC2CCC1C1CN(C(c3cc(C)sn3)=O)CC21 C1(C(N(C)Cc2scc(C)c2)=O)CCN(C(=O)NC2(C)CC3CC3C2)CC1 c1(C(=O)NC(C)(C)CNC(c2[nH]ccc2C2CC2)=O)cc(F)cc2c1CCC2 c1(C(=O)NC(CNC(CN(C2CCC2)C)=O)C2CCC2)ncccc1N c1(CC)cnc(O)c(C(=O)NCCCN(C(=O)CCC2CCCCC2)CC)c1 Cc1cccc(C(=O)NC2CCN(C(=O)C=Cc3nc(C)c(C)[nH]3)CC2F)c1Cl C1(C(N(C)Cc2cnn(C)c2)=O)CC(O)CN1C(=O)C=Cc1cn(C)cn1 N1(C(C(Cc2ccoc2)NC(=O)CCN2CCOCC2)=O)CCC(F)(CF)C1 C1(C(C(N2CCC(CNC(CSC)=O)C2)=O)C)CCC(C)(C)CC1 C(CN=C(NCc1cc(C)cnc1O)NCC1CCOC1=O)OCC=C N1(C(CN2CCC(C)CC2)=O)CCC(C)(C)C(NC(=O)CC(F)F)C1 CC1CCCC(=O)CN1N1CC2C(c3ccccc3)S(=O)(=O)C2C1 Cc1cc(C(=O)NC2CCC(NC(c3cc(N)cc(O)n3)=O)C2)c2occc2c1 N1(CCCCCNC(C2CC23CCC3)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC1 N1(C(C(C)(C)CF)=O)CCC2(CC1)CC(NC(=O)C(F)CC1CCCC1)C2 C1(C(=O)NCC(C)C(=O)NCC(c2cccnc2)C)CC2(CSC2)C1 CC1CON(C(=O)CC2CC(=O)C2)CCN1C(=O)CC1CC1.N12CC1CCC2=O N1(C(N(CCO)CC2CCN(CC)CC2)=O)CC(C)N(CC)C(C)C1 C1(NC(C)=O)CCN(C(=O)CCc2ccncc2)C1(C)C.c1(CC)ccc(F)cc1 C1(NC(c2[nH]cc(C)c2)=O)C2CC3CN(C(=O)CC4CCC(O)C4)C1C3C2 Cc1nc(C=CC(=O)NC2CCN(C(C3(C)CCC(C)CC3)=O)CC2F)[nH]c1C c1(C(F)(F)F)ccccc1.C1(N(C)CC)CC(N)C1.C1(C)CNC(=O)N1 N1(C(C(=Cc2cccs2)C)=O)CC2(CC(NC(c3oc(CO)cc3C)=O)CO2)C1 C12(C(N(CC(F)F)CC)=O)CC(C)(CN1C(C1CC1C1CCCO1)=O)C2 c1(CC(=O)NCC(CCC)Cc2ccccc2)ccc2c(c1)CCC2.C1(=O)CO1 C(=O)(CCCCC(C)(C)C)N1C2CC(CNC(C(C(CC)(C)C)O)=O)C1CC2 N1(C(c2c(C)cc(C)o2)=O)CC(NC(c2cccn2C2CCCC2)=O)CC(C)C1 C1(OC)CCC2(CCN(C(=O)C(C)(CSC)NC(C3CCCC(C)(C)C3)=O)C2)C1 c1(C(=O)NCCNCCO)cccc2ncccc12 Cc1nc(C(C)C)ncc1C(=O)NCC1CCCCN(C(=O)C=CC2CCC2)C1 N(C(=NCCCN(C)C1CC1)N(C)C)CC(N1CCOCC1)C(C)C C1(C(N2CC(C)CC(CC)C2)=O)CCN(C(c2cc(O)n(C)n2)=O)CC1(C)C N1(C(C2(C3CCCO3)CCC2)=O)CCC(NC(=O)C(C)=CCOC)C(F)C1 C12(NC(=O)C3CC3)CCCC1N(C(=O)COc1c(OCC)cccc1)CC2 C(=O)(CCC(=O)NCC1CC(C)N(C(c2ccc(Br)o2)=O)C1)N(CC)CC C(C)(C(=O)NCC(O)CN(C)C(c1cnc(C)nc1)=O)(C(C)C)OC C(=O)(CC(COC)NC(c1cc(C#N)cs1)=O)Nc1cn(CCC#C)nc1 N1(C(C(c2c(C)cccc2)C)=O)CC2CC(C1)N(C(=O)C=CC(C)=O)C2 CON=C(C(=O)NC(C)CNC(c1cncc(Cl)c1Cl)=O)c1ccco1 C(=O)(C1CCc2ccccc21)NCC1(O)CCN(C(C2(CCN(C)C)CC2)=O)C1 C(=O)(C(C(=O)NCC1CCCN(C(=O)CCc2cncc(F)c2)C1)OC)OCC N1(C(CN(C(c2ccc(C)s2)=O)CCO)=O)CC2(CCN2C(C2CC(C)CO2)=O)C1 CC1CN(C(=O)CN2CCC(C)(C)C2)CCC1NC(=O)Cc1cccc(Cl)c1 C1(NC(C2N(C(C)=O)CCC2)=O)CN(C(C2OCC2(C)C)=O)CC2(CCC2)C1 C(C)(CNC(=O)C(C1CCOCC1)OC)(C(C)C)NC(CCC=CCC=C)=O C1(NC(C2C(C)OCCC2)=O)CCCCN(C(c2cc(O)cnc2N)=O)C1 N1(C(c2c(C(C)C)nns2)=O)CC2CCN(C(c3ccoc3Br)=O)C2C1 C(C(C(=O)N1CCCC(C)(CC2CC2)C1)C(C)C)NC(Cc1nc(C)[nH]n1)=O c1(C(N(C(C(=O)NCC(C)C)C)C)=O)ccc(NC=O)cc1 c1(OCCNC(C(N2CCCCC2)C2CC(OC)C2)=O)c(F)cccc1F CCCS(=O)(=O)C(C)C(=O)N1CCOCC(NC(C2(CN(C)C)CCCC2)=O)C1 c1(CC(=O)NCC2(O)CCN(C(=O)Cn3ncnn3)C2)cccnc1Cl N1(C(=O)OC(C)(C)C)CC2CCC(=O)NC2C1.c1(CC)ncc2cc1NC2=O N1(C(c2ccc(CC)c(C)c2)=O)CCCN(C(C2CCN(C(C)=O)C2)=O)CC1C O=c1cc(N2CCC23CC(CF)C3)nc2ccccn12 CCC(C)(CNC(=O)CCC1CC1)C(=O)NCC1(OCC)CC1 N1(C(C2C(C)OCC2)=O)CC2(CCCC2NC(C2C3CCCOC23)=O)C1 CC(C)CC(O)C(=O)NC1CC(C)(C(=O)NC(c2ncc[nH]2)CO)C1 C(C(COC)CC(=O)NCCN(C(=O)C(C)(F)CC1CCCC1)C1CC1)OC C1(C(N2CC3C(CNC(Cn4cc[nH]c(=N)c4=O)=O)C3C2)=O)CN2CCN1CC2 N1(C(C(CC)NC(N)=O)=O)CCC(NC(=O)C(c2ccccc2OC)O)C(F)C1 c1(C(=O)NCC2N(C(C3N(C)COC3)=O)CC2)c(F)ccc(Cl)c1F N1(CCC2(NC(c3ccc(OCCC)cc3)=O)CC2)C(C)(C)CC(=O)CC1(C)C C1(C(=O)NCc2occ(C)c2)C(C)OCCN1C(C1COCC(C)O1)=O N1(C(CCCN(C(C)=O)C)=O)CC2CCC(C(N3CCCCC3C(C)C)=O)(C2)C1 C1(C)(C(=O)NC2CC(C)(CNC(Cn3cc(C(C)O)nn3)=O)C2)CCC(=O)N1 C(=O)(C1CC=Cc2ccccc21)NCC(C)NC(c1c(N(CC)CC)nccc1)=O Cc1ccc(O)c(C(=O)NC2CC3CC2CC3C(N2CCC(C)(F)CC2)=O)c1 N1(C(CN(C(COCCC#C)=O)CCOCCO)=O)CC(COC)CC1C CC(F)(C(=O)NCc1ccoc1C(=O)NCC1CCC2CC12)c1ccon1 N=c1nc(O)c(C(N2CCCCC(NC(=O)CC3COC4CC3C4)C2)=O)c[nH]1 N1(C(C2(CCCC)CC2)=O)CC2(CNC(=O)COC)CC1CO2 C1(C(=O)NCCCN2CCC(N(C)C)CC2)CCCCC12CC2(F)F c1(CC)cccc(C(=O)N(CCN(C(=O)Cn2nc(C)oc2=O)C)C(C)C)c1F CCCCCCC(O)CCC(=O)N1CCC2(CC(NC(=O)Cc3cnc[nH]3)C2)C1 C1(CCC(=O)NCCN(C(C2CCC2F)=O)CC2CC2)CCCCC1 N1(c2c(CNCC=COc3ccc(OCC)cc3)cccc2)CC(C)OC(C)C1 CCC(CC(=O)NCC1CC1NC(=O)COCCN(C)C)C(F)F C1(COC)(NC(C2CCCS2)=O)CCCN(C(C2CCCCC2(C)C)=O)C1 N1(C(c2ncc(C(F)(F)F)cc2Cl)=O)CCCC(C2CN(CC3(CO)COC3)C2)C1 c1(C(=O)NCC(=O)N(CC(C)NC(CC(=O)OC)=O)C)cc(F)cc(F)c1 CC1SCCN(C(C2(NC(=O)Cn3cnnn3)CC(O)C2)=O)C1C C1(NC(CSCC)=O)CC(NC(c2cc(C3CC3)ccc2C)=O)C12CCOCC2 CC#CCCCC(=O)N1CCOCC1CCCNC(=O)COC1(C)CCC1 c1(CC)cc(C(N2CC(CNC(=O)C=C(C)C3CC3)C(C)C2)=O)cc2c[nH]nc12 CCC(O)C(C)C(=O)NC1(COC)CCN(C(c2ccc(F)cc2C)=O)CC1 c1(C(N(CCNC(C2CCC(CC)C2)=O)C)=O)ccc(C2COC2)cc1 C(=O)(C1=CCCOCC1)NC(CNC(C(=CC1CCCC1)C)=O)C c1(C(N2CCC(O)C(C(N3CCOC4CC34)=O)C2)=O)cc(F)c(F)c(F)c1 c1(C(N2CCN(C(COC)=O)CC2c2cn[nH]c2)=O)ccn2nnnc2c1 c1(C(N2C(CNC(c3c(C)cno3)=O)C(C)CC2)=O)cn(C)c2ncccc12 c1(C(=O)NCC2(CCCNC(c3cc(F)cs3)=O)CCCC2)cnn2c1OCC2 C1(CNC(C2C(C)C2C)=O)CN2CCCCC2CN1C(=O)CCc1nccs1 C1(NC(C2C(C(C)C)CCC2)=O)COCCN(C(=O)C(F)C(C)(C)O)C1 C(=O)(C(CNC(c1csc(CSC)n1)=O)C(C)(C)C)NCC C1(C)(CNC(c2c(C)ncs2)=O)CN(CC2CCC(F)(F)C2)CCO1 CCCC(CCCNC(=O)CCOCC(F)(F)F)NC(=O)CN=S(C)(C)=O O=C(CCC(=O)NC1CN(C(c2ccco2)=O)CC1O)Nc1nccs1 c1(C(N2CC(CCC)N(C(=O)CCN(C)CCC)CC2)=O)cc(O)cc(N)c1Cl C1(CC)C(NC(=O)CC(C)(C)CC)CCCN1C(c1coc(CC2CC2)n1)=O C1(NC(C2ON=C(C(C)C)C2)=O)CC2CCC(C1)N2c1ncnc(O)c1Br S(=O)(=O)(c1cccc(Cl)c1Cl)NCC12C(CN(C(C(C(CC)C)N)=O)C1)C2 CC1(C)CC(C(=O)NC2CCC(C3CC3)C2)CN(C(=O)C(=O)NCC2CC2)C1 C1(OC)CN(C(=O)C(CNC(=O)CCCc2cnn[nH]2)(CC)CC)C2(CCC2)C1 C1(NC(C(COC)O)=O)CC12CCC(NC(c1c(C)ccnc1C)=O)CC2 C(=O)(C1=CCCCC1C)N1CC(OCC)C(CNC(c2cnc[nH]c2=N)=O)C1 C1(C(=O)NC2CN(C(c3cc(CC)n(CCO)n3)=O)CC2C)CCC(=O)CC1C C#CC1CCC(C(=O)N(CCOC)CCNC(=O)CCC2CCCN2C)CC1 C1(C)(OCC(=O)N(C(CO)CO)C)CN(C(=O)C(F)n2ccnc2)C1 C1(C(N(C)CC2CCN(C(COC(C)C)=O)C2)=O)Cc2ccccc2N(C)C1=O C(=O)(C1=COCCC1)NCC(CC)NC(c1cc(-c2ccccc2C)[nH]n1)=O CC(F)(F)C(F)(F)CCS(=N)(=O)Cc1nc2ccccc2n1C(F)F Cc1ccc(CCC(=O)NCC(C2CCCC2)NC(C2CC2C#N)=O)cn1 c1(OC)ccc(C(=O)NC2(c3ccccc3)CN(C(=O)C=C(Cl)Cl)C2)cc1SC C(=O)(C(CC(F)F)NC(C1C=CCCC1)=O)NCc1ccc(=N)[nH]c1 n1(C(CC)(C)C)nnnc1C(c1cnc(C2OCCO2)o1)NC(C)C1CC1 C(=O)(C(C)(C)CC#N)NC(c1ccc(CNC(C2(C(F)(F)F)CC2)=O)cc1)C Cc1nc(O)nc(O)c1CCC(=O)NC1CCN(C(=O)CC(C)C(F)F)C(C)C1 C(=O)(CCCCNC(=O)C(C)(C)C1CC1)NC1C(CN(C)C)C1 c1(OC)ccc(C)c(C(N2CC3(CCN(C(=O)CCc4cnco4)C3)C2)=O)c1N NC(=O)CC(O)C(=O)NC1CC(CC(=O)NC(CCO)C2CCC2)C1 c1(N(CC(C)C)C)ccc(NCCNC(=O)Cc2cc[nH]n2)cn1 C1(C(=O)NCCC#CCC)CCN(C(c2sccc2C)=O)C12CC2 C1(CC(N2CCC(C)(CNC(CN(CC)CC)=O)C2)=O)COc2ccccc2O1 c1(NC(C2(C)N(Cc3c(SC)cccc3)CC2)=O)cc(Cl)c(Br)cn1 C1(C(N)=O)CN(C(=O)C(C2CC2)NC(=O)Cn2cncn2)CCO1 c1(C(N2CC3(N(C(CCOC)=O)CCCC3)C2)=O)oc2ccccc2c(=O)c1C Cc1[nH]nc2c1CC(C(=O)N(CCCNC(=O)C(C1CCCCC1)F)C)CC2 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)OC(CC(C)CN(C)C)=O Cc1ccc(C(=O)NCC2(CNC(=O)Cn3nnnc3C)CC2)c(F)c1 CCC(CNC(c1cc(COC)oc1C)=O)(CC)NC(C1C(COC)C1C)=O N1(C(c2ncccn2)C)CCCC(NC(c2ccccc2C#N)=O)CC1 C1(NC(=O)OC(C)(C)C)CCC12CN(C(=O)NC1CCCN1c1cccnn1)C2 c1(C(=O)NC2CCCC(NC(CCC=C=C)=O)C2)ccc2c(c1)CNC2=O N1(CCN(C(C(C(N(C(COCCC)=O)C)CC)N)=O)C)CC2CCC1C2 Cc1cn(C)cc1C(N1CCC(C2CCCCN2C(c2oncc2C)=O)C1)=O c1(C(N2CCC(CCN(C(C3C(=C)C3)=O)C)CC2)=O)sc2ccsc2c1C CC1CN(C(=O)C=CC(C)(C)C)CCC1NC(=O)CCCN1C(=O)CN(C)C1=O N1(c2scc(C)n2)CCC2(CC1)CC2C(N1CCCC(O)C1C)=O c1(C(N2CCC(CCNC(C3C(OC(C)=O)C3)=O)C2)=O)cc(C(F)F)ccc1F CC(C)C(C(=O)NCCC1CC(NC(=O)COC2CCOC2)C1)NC=O CN(C1OCCc2sccc21)C(c1cc(Br)c(Cl)s1)C(=O)NC(C)(C)C c1(C(N2CCCN(C(C(CC(C)C)O)=O)CC2)=O)ccc(C#CC2CC2)cc1 CCCC(C(=O)N1CCC(NC(c2ccccc2N(C)C(C)=O)=O)C1)OCC N1(C(C2(F)C(C)OCC2)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C1=NOCC1 C(=O)(C(O)CC(F)(F)F)N1CC(C)C(C)(CNC(c2ccc(=O)n(C)n2)=O)C1 N1(C(C(C(C)C)SCC)=O)CC(CO)C2(C1)CN(C(=O)Cc1ccccc1F)C2 c1(C(N2CC(C(C)C)N(C(=O)C(F)C3CCC3)CC2)=O)csc(S(N)(=O)=O)c1 C=CC(F)(F)C(=O)NCCCSC.N12C(CC1C)CC2=O Cc1nc(CC(C)C)c(C(=O)NC2CCC(NC(=O)Cc3csc(C)n3)CC2)s1 C1(C(=O)NCc2cc(CC)no2)N(C(=O)C(N2CCOCC2)C)CC12CCCC2 C1(C(N(C)CC2CCCC(CC(F)(F)F)C2)=O)CCCN(CC(=O)O)C1=O C=CC(C)(CC)C(=O)N1CCN(c2cccc(CN3CCS(=O)CC3C)c2)CC1 c1(C(=O)NC2(CC3CC3)CC2)n[nH]c2c1CN(C(C1CCC1)=O)C2 c1(C(N2CCC(N(C)C)C2)C(=O)NCCSC)cc(F)ccn1 C1(NC(CCC(=O)N(CCC)CC)=O)C2CCC1N(C(=O)CSc1cccs1)C2 CCCCC(C(=O)NC(CCF)C(=O)OC)NC(=O)CCSCCCC n1(CC)nc(C(=O)NC2CN(C(=O)C(F)(F)CC3CC3)CC2O)c(Br)n1 c1(C(=O)NC(C2(CNC(C3CCC=CCC3)=O)CC2)C)noc2c1COCC2 CCC(COC(C)C)(C(=O)NC(c1cc(F)ccc1Cl)C(=O)O)c1ccccc1 Cc1ccc(Br)c(F)c1C(=O)NC1CCC(O)C1 N1(CC)N=C(C(=O)NCC2(NC(c3nc(Cl)cc(N)c3Cl)=O)CC2)CCC1=O c1(C(=O)NCC2N(C(c3occ(C)c3)=O)CCC2C)cc(F)c(C)c(N)c1F N1(C(c2ncc(C)cc2C)=O)CC(C)CN(C(=O)CN(C(=O)C(C)C)C)CC1C C12(NC(c3nc(Br)c[nH]3)=O)CCN(C(c3cccc(F)c3F)=O)CC1C2 c1(C2N(CCC)CC2(C)C)ccc(C(C)C)cc1 C1(NC(C2CC(=O)NC2)=O)CCN(C(=O)CCOCC2CCCO2)CC1F C1(C(N2CCC(OCCNC(C=CC(CC)C)=O)CC2)=O)CN2CCN1C(C)C2 c1(N2CCC(C)OCC2)nc2c(c(=NC(C)c3cn(C)nc3C)[nH]1)SCC2 Cc1cc(C(=O)NC2CC(NC(C3(CF)CCOCC3)=O)C2)ncc1Cl C1(C(=O)NCC2C(C)(C)C2(C)C)(CC)CCCN(C(=O)CCNC(C)=O)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1(CN(CC(C)(C)S(C)(=O)=O)C)CCC1)N CN=C(NCc1cc(C)ccc1O)N1CCN(CC2CCOC2=O)CC1 Cc1cc(C(=O)NCCN2CCN(Cc3cnn(C)c3F)CC2)ccc1C(=O)O C1(CNC(CSCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CCCO1 c1(C(C)=O)ccncc1NC(C1CSCCN1C(=O)C(C1CC1)N(C)C)=O C1(OC)CCC(C)(C)N(C(=O)C(=O)N(C)CC2CCC23CCC3)C1 N1(C(C23C(CCN(C(CC(C)C)=O)CC2)C3)=O)CCC(F)(F)C(F)C1 C1(C(=O)OC(C)(C)C)CC2(CCC2OCC)C1.C12CCCN1C2=O c1(OC)cnc(C(N2CC3C(CNC(=O)Cc4sc(C)cc4C)C3C2)=O)nc1 c1(C(N2CC(CCNC(C)=O)OCCC2)=O)ccc2ncn(C)c(=O)c2c1 N1(C(C2CCSCC2)C(=O)NC(CC)C)CCOC2(CCC(C)(C)C2)C1 Cc1[nH]nc2c1CC(C(N1CCN(C(c3nnn(C)c3N)=O)CC1CF)=O)CC2 C1(CNC(CCC(=O)N(C)C)=O)COC(C)(C)CN1C(=O)C(CCS(C)=O)N(C)C C(=O)(C1CCCc2nn[nH]c21)NC1CN(C(C#CC2(C)CC2)=O)CC1O c1(C(N(C2CCN(C(=O)C(F)=CC3CC3)C2)CCC)=O)cc(C(N)=O)co1 C(=O)(CCC1CCc2ccccc21)N1CC=C(CNC(c2c(C)non2)=O)CC1 C1(O)(CCNC(c2nn(C)c(C3CC3)c2)=O)CCCN(C(c2ccsc2Cl)=O)C1 C(C(=O)N(C)CCNC(=O)CC(F)(F)Cl)(C(C)C)c1cnc(C)s1 C1(C(=O)NC2CCCC(O)C2)CC1C1CN(C(=O)C(F)(F)C2CC2)C1 C#CCC(CC#C)C(=O)NCC1CC(OC)CN1C(c1sccc1C)=O C1(C(=O)NCCCNC(C(c2nc(C)sc2)=O)=O)CCC2C1C2(F)F c1(C(=O)NC(C)CNC(=O)C(c2cncn2C)C)ccc2c[nH]nc2c1 C1(NC(C2C(OC)C2)=O)CC2(CCN(C(c3ccc(-c4cc[nH]n4)cc3)=O)CC2)C1 c1(N(C(C)C)C)ccccc1NCC(N1CCN(CC(=O)O)CC1)=O N1(C(c2ccc(C)nc2)=O)CCCC(O)(CN(C)C(c2cc(O)nc(Cl)c2)=O)C1 N1(C(CNC(CC)=O)=O)CC(CNC(c2cncc(SC)c2)=O)CCC1C c1(C(=O)OC)nc(=NC2CN(C(C3CC3Cl)=O)CC3(CCC3)C2)cc[nH]1 c1(N2Cc3c(CNC(CC(C)(C)OC)=O)cnn3CC2)cc2n(n1)CCCC2O c1(C(=O)NC2CCC(O)CN(C(C3C4CCCC34)=O)C2)cc2ccnc(Cl)c2[nH]1 c1(CC)cc(C)ccc1C(=O)NC1(CO)CN(C(=O)C(F)(F)C(O)C2CC2)C1 c1(CNC(c2ccc(-c3ccccc3)o2)=O)ccc2cc(C(F)(F)F)ccc2c1 c1(C(=O)NCC(C)(C)CNC(C2CC3(C2)CC3F)=O)ccc2oc(O)nc2n1 c1(CN2C(COC)CN(C(C3(F)CC3)=O)CC2)c[nH]c2ncc(Cl)cc12 NS(=O)(=O)c1ccccc1-c1cc(-c2ccncc2)ccn1 CCC(CC(=O)NC1(C)CCN(C(=O)C(C)Oc2cccc(F)c2)CC1)C(F)F c1(C(N(CC(C)CNC(C2CCC(C)O2)=O)C)=O)cc2ncccc2cc1Cl N1(C(C(C2CC2)OC)=O)CCN(C(C2(Br)CC2)=O)CC1CCO Cc1ccc(CC(=O)NCC)cc1.C12(CCOC1)C(=O)O2.C1(=O)CN1.C(C)(C)(C)NC c1(C(N2C(c3ccn(C)n3)C(C)(C)C2)=O)c[nH]c2ccc(I)cc12 N1(C(C=CC=CCC)=O)C2CCC1C(F)C(NC(c1ccc3c(c1)OCC3)=O)C2 c1(-c2scc(C)c2)ccc2c(c1Oc1ncccc1C1CC1)OCO2 N1(C(C2N(CC)CCC2)=O)CCC2(CC1)CCN(C(=O)Cn1ccccc1=O)C2 C123CC1CN(C2)C3=O.c1(NC(C(c2ccc(F)cc2)OC)=O)cc(O)ncn1 c1(OCC#C)ncccc1C(=O)NCC1(CNC(c2[nH]ccc2C)=O)CCC1 c1(C(=O)NCC(CC(C)C)NC(c2cnc(C)[nH]2)=O)cc2n(c1)CCCNC2=O c1(C(=O)NC2C(NC(C(C(C)C)SCC)=O)C2)cc(C)c(F)cc1Cl C1(C(N(C(C)(Cl)Cl)CCC#N)=O)CCCCN1C(c1c[nH]c(=N)s1)=O C=C(C)CN=C(NCc1c(C)cc(C)cc1C)N1CCCC(C)(C#N)C1 c1(C(=O)NC(CN(C(=O)CN2C(=O)CNC2=O)C)(C)C)ccnc(Cl)c1N C(CCN=c1[nH]cnc(Cl)c1Br)N(C(c1cc(C)c(Cl)cc1)=O)C C1(C(N2CC(C#C)(O)C2)=O)CCN(C(c2coc(C(N)=O)c2)=O)CC1(C)C Cc1cc(C(N2CCC(N(C(=O)CCc3cccc(O)c3)C)C2)=O)ncc1F c1(C(=O)NC23C(CN(C(CCOC(C)C)=O)C2)C3)ccc2c(c1)NC(=O)C(C)O2 C1(CNC(c2cnc(C(C)OC)s2)=O)CCCCCN1C(c1ccc[n+]([O-])c1)=O c1(OC)ccc(CCCNC(=O)CCC2CCCN(CCC(C)C)C2)cc1OC C(=O)(C(C)(C(C)C)OC)NCC12OCC(NC(CCN(CC)CC)=O)(C1)C2 c1(CC(N2C(C)(CNC(COCCC=C)=O)CCC2)=O)ccc(F)c([N+](=O)[O-])c1 CN1CCC(O)(CNC(=O)CC2CN(C(c3ccc(C(N)=O)[nH]3)=O)CCO2)C1 O=C(CC1OCCc2ccsc21)N1CCCC1C(c1ccccc1)O c1(NC(C(C2CCCN(C(C(C3CCCC3)OC)=O)C2)C)=O)cccc(F)c1C c1(CCN(C(C2CCN(CCO)CC2)C(=O)O)C)ccc(O)c(OC(F)(F)F)c1 c1(C(=O)Nc2ccc(NC(c3c(C)c[nH]c3)=O)c(F)c2)ccc2oc(C)nc2c1 N1(Cc2sc3ccccc3c2)CCOC2(CCC(C(F)(F)F)CC2)C1 c1(C(N2C(C)CC(CNC(C3(S(N)(=O)=O)CCC3)=O)C2)=O)cccc2c1OCO2 CC1CCC1CNCCNC(C1(NC(=O)C(N2CCCC2)C2CCCC2)CC1)=O CCCC(C(O)C(=O)NCCCOC(=O)NC)NC(=O)C(N1CCOC1=O)C c1(CC)cc(C(=O)NCC(C2CC2)NC(c2cc(F)n[nH]2)=O)c(C)nn1 C1(C2(O)CCOCC2)(C(=O)NCCCC(C)NC(CCC(C)SC)=O)CC1 c1(CCC)cc(C(N2CCCCC2CNC(=O)CC23CCCC2C3)=O)n(C)n1 c1(C(C)NC(=O)C=C2CCC2)ccc(CNC(=O)CCN2CCCCC2)cc1 CC(C)C(O)C(C)C(=O)N(CCC(=O)Nc1cccc2c1OCO2)C(C)C N1(C(C(C(C)OC)N(C)C)=O)CCOCC(C(=O)NCCCn2nccn2)C1 n1(C(C)C)ncc2c1CC(NC(N1CCCCCCC1C)=O)CC2 C1(NC(C2(N(C)C)CC2)=O)C2CN(C(C3CC(n4ccnn4)C3)=O)CC12 C(=O)(CS(=O)(=O)CCO)N1C(CNC(C(C)CC2CC2)=O)CC(O)C1 c1(C(=O)NC(C2CCCC2)CNC(c2[nH]cc(C(C)=O)c2)=O)nc(F)ccc1Cl C1(NC(C2(C(=O)NC)CC2)=O)CC2(C1)CN(C(c1nn(C)c(Cl)c1Cl)=O)C2 c1(CC)ccc(C)c(C(=O)NCC2CN(C(=O)CCN(CC)CC)C2)c1 CC(C)CC(O)C(C)C(=O)NCCCNC(=O)CCc1cc(F)cc(F)c1 c1(OCCC(=O)NCC2N(C(CN3C(C)CC3)=O)CCOC2)cccc(Cl)c1Cl c1(C(=O)NC(C)(C)CNC(=O)C(n2ccnn2)C2CC2)ccc(CO)s1 CCC(C)(C)CCCC(=O)N1CCN(C(c2scc(C)c2C)=O)C(CO)C1 C1(CNC(COC2(C)CCC2)=O)CCCC(CNC(=O)CC2CC3(CC3)CO2)C1 C1(O)(CC(=O)NC2CCCC(CO)C2)CCN(C(C2(C(N)=O)CC2)=O)CC1 CC(Cc1cn[nH]c1)CN=c1[nH]c(=NCc2nnc3n2CCOC3)c2sccc2[nH]1 C1(CNC(c2c(CC)scn2)=O)CN(C(c2nc(OC)ccc2Cl)=O)CCC1C c1(-c2c(OC)cc(C(=O)Nc3sncc3C#N)nc2)c(C)cc(C)cc1C C1(C)(CNC(C(=O)NCC)=O)CN(C(=O)C(C)OC2CCOC2)CC1C Cc1c(F)cc(C(N2CCC3(CC(C(N4CCCCC4C)=O)C3)C2)=O)cc1Br N1(C(C2(COC)CC2)=O)CCN(C(=O)CC2OCCC2(C)C)C(C2CC2)C1 C1(NC(Cn2cc[n+](C)c2)=O)CCCC(CNC(=O)C(N)=O)C1 Fc1cccc2ccnc(N3CCN(Cc4cn[nH]c4)CC3)c12 C=CCC(C(=O)N1CCCC1(C)CCC(=O)Nc1cn(C)nc1O)C(C)C c1(-c2nn(-c3cnc(C)s3)c(-c3cc(F)c[nH]3)n2)c2ccccc2nn1C c1(OCC(=O)NCC2N(C(CCc3nc(C)sc3)=O)CC=C2)cccc(F)c1F C1(C(=O)NCC2CC(NC(CC3C(C)=NNC3=O)=O)C2)CC2(CCO1)CC2 C1(C(N2CCC(NC(=O)Cn3ccc(Br)n3)C2)=O)CC2(CCC2O)C1 C1(CC(N2C(COC)CCOCC2)=O)CCCCC1(F)F N12CCN(C)CC1C(C(=O)OC)N(CCC#N)CCCCC2=O.C(CC#N)N.CS N1(C(C(=O)Nc2c(C)nc(Br)cc2)=O)CCCC(C)(C)CC1 c1(NC(C(=O)NCC2CCC(C#C)CC2)=O)ccc2cnn(CC)c2c1 c1(CC(C(=O)NC(C)(C)CNC(=O)C=C(Cl)Cl)NC(=O)OC)cccc(F)c1 Cc1nc(C(=O)NC(C)CCCNC(C2CC2Sc2ccccc2)=O)c(C)o1 C1(NC(c2n(C)nc(C)c2Cl)=O)CCCC2CN(C(C3CCCN3C=O)=O)CC12 C12(NC(CCN(CCC)C)=O)CCC(CC1NC(C1CC(n3ccnc3)C1)=O)C2 C1(C(N(C)CCc2cnc[nH]2)=O)CCC(O)CN1C(c1sccc1F)=O Cc1sc(Cl)c(C(=O)NCc2cn(C3CCN(C(=O)C(C)O)C3)nn2)c1C Cc1c(NC(=O)CCC(C)N(C)C)cnn1C1CCOCC1 C1(C(=O)NCC(C)SC)CCN(C(=O)CC2(O)CCCCC2)C(C)(C)C1 C(=O)(CC(C)CCC(=O)NCC(C(N1CCC(C)(NC(=O)NC)C1)=O)C)NCC N(C1c2ccccc2CCC1F)C(c1c(C)cc(Cl)nc1N)=O C#CC1(C)CCCN(C(c2cc(C3CCC3)on2)C(=O)NC2CCCCCC2)C1 C(=O)(C1=CCCC(C)(C)C1)NCC(C)(CO)NC(CC(C)P(C)(C)=O)=O C(CCC1CC1)(C(=O)NCC(=O)NC1CC1)N1C(CCO)CCC1.C1(CS)CCCCO1 c1(N2CCC(COC)C2)nc(NC2CCCc3occc32)c2c(n1)c(C)nn2C c1(C(=O)OC)ccc2nc(N(C)C3CC3)[nH]c(=NCc3ccc(F)cc3I)c2c1 C1(C(=O)OC(C)(C)C)CC(F)(F)C1(F)Cl.C(=O)(C(=O)OC)N(C)C c1(C(=O)NC(c2c(F)cccc2F)c2cccc(C)c2)cnc2sc(C)cn12 C1(CC(=O)NCCC2CN(C(C3C(CCC)C3)=O)C2)CCCC(O)C1 C1(C(N(CC(C)NC(C2=C(C)OCCS2)=O)C)=O)CCCC2CCCCC12 C(CCCCCNC(C1(CO)CCCO1)=O)NC(c1cc(COC2CC2)on1)=O CC1CN(C(=O)CCCF)CCN1C(c1ccc(O)c(Br)c1)=O C1(C(C)NC(=O)CCc2nncs2)CCCCN1C(=O)CCc1cnn(C)c1 c1(C(=O)NCC(C)CNC(c2cccc(N)c2Br)=O)cc2ccncc2s1 c1(C(=O)NC(CNC(C=C(CCC)C)=O)C2CC2)ccn2ncc(Br)c2n1 c1(C(C(=O)NCC(=C)C)N(C(C)C(C)(F)F)C)ccc(Cl)c(F)c1F c1(C(N(C2CCNCCC2C)c2ncc(C)nc2)=O)c[nH]c2ccc(F)cc12 N1(C(C2C(NC(C3(OC)CCCC3)=O)CCOC2)=O)CCN(C)C(=O)C1 CN1CCC2CCN(C(=O)CC3CCN(C(c4ccc(O)cc4)=O)CC3)CC12 N1(C(C(C(C)C)N(C)C)=O)C(CC(=O)NCC(F)(F)CC2CC2)C2CCCC12 C1(NC(C2N(C(N)=O)CCC2)=O)C2CN(C(c3cnn(CC4CC4)c3)=O)CC12 C1(C#N)(C(N2CCCN(C(C(C)Cc3cnc[nH]3)=O)CC2)=O)CC2(CCC2)C1 CC(C(=O)OC(C)(C)C)C(=O)NC1CCCN(C(c2cnc[nH]2)=O)C1 c1(OC(C)C)cc(Nc2nc(Cl)cs2)c(-c2ccc(ON3CCCC3)c(O)c2)cn1 CN1CNC(=O)C12CN(C(=O)CCC1CCCCN(C(C3CC3(F)Cl)=O)C1)C2 c1(CC(=O)NCCCN(C(CN2C(C)CCC2)=O)CCO)cc(Cl)n(C)n1 c1(C(N2C(C)C(NC(c3coc(Br)c3)=O)CCC2)=O)nc2ccccn2n1 N1(C(C(C)(F)F)=O)CC2(CC1CNC(=O)COC1CCCCCC1)CC2(F)F c1(C(N2C(CN(c3ncc(C#N)cc3Br)C)CCC2)=O)cccc2c1nnn2C C(C(C)(C)CC(=O)NCc1csc(CNC(c2cc(C(C)C)nn2C)=O)n1)OC c1(C(=O)Nc2cc(F)cc(C(F)(F)F)c2N)ccc(F)c2occc12 C1(CC)CCN(C(C2(O)CCOCC2)=O)C1C(=O)NCc1csc(C)n1 c1(OC)c(C)cc(C(N2CCN(c3ccc(F)cc3)CC2)=O)cc1Cl C12(NC(c3ccc(C(F)F)cc3F)=O)CCC(C1)N(C(C1CCCCS1)=O)C2 C1(C(CNC(c2nc(C)sc2)=O)F)CCN(C(=O)CC(O)c2ccccc2)CC1 N1(CC(=O)Nc2cccc(-c3nn[nH]n3)c2)CCc2c(O)cc(O)nc2C1 Cc1ccc(C)c(C(=O)NCC(C)(C2CC2)NC(=O)CCc2ccn(C)n2)c1 C#CCC(O)C(=O)N(C1CC1)CC1CCCN1C(c1cnc(C2CC2)nc1)=O N1(C(c2n(CCCC)ncc2)=O)CCCC(NC(=O)CCc2ncnn2C)C1C c1(C(=O)NC2C(C)N(C(=O)CCCC3CCC3)CCC2)cnc2ccccc2n1 C(=O)(C1=NOC(C)(C)C1)N1CCC(CC(C)NC(=O)C(C2CCOCC2)F)CC1 c1(CC(=O)NCC(CN(C(C(CC)O)=O)C)O)c[nH]c2cccc(Br)c12 c1(OCC(=O)N(CCNC(c2c(C(C)C)nns2)=O)C)ccc(F)cc1F C(=O)(C1=NOCC1)NC(COC(C)C)C(=O)NC1(F)CCN(C)C1 N1(C(c2cnc(C(C)C)s2)=O)CC2(CCCC2NC(=O)CC(C)P(C)(C)=O)C1 c1(CC(=O)NC2C=CC(CC(=O)N(C(C(CC)C)C)C3CC3)C2)ncccc1F c1(C(N2CC(C)N(C)C(=O)C2)C(=O)NCC2CCCO2)cnc2ccc(Cl)cn12 c1(OC)c(F)cc(CN2CC3CCN(C(C4(C)CCCN4)=O)C3C2)cc1F c1(C(=O)NCC2(NC(C(c3c(C)n[nH]c3C)C)=O)CCC2)cc(Cl)c(F)cc1Cl CC1(C)CCN(C(c2ccc(N)c(F)c2)=O)C1CNC(=O)CCN1CCC1 CCC(C)CCC(=O)NC1CN(C(c2cc(N)ccc2C)=O)CC1SC C(=O)(C(CO)C(C)(C)C)NC1C2(C(=O)NCC(C3CCC3)OCC)C3CC1CC23 c1(C(N2CCOCC(NC(c3cnn[nH]3)=O)C2)=O)cc(Cl)c(Cl)c([N+](=O)[O-])c1 N1(C(C(C(C)C)n2ccnc2)=O)CC2CCN(C(c3sccc3C#N)=O)CC2C1 Nc1c(C(=O)N(C2CCN(C(C34CCC3C4)=O)CC2)CCO)ccc(Cl)c1F N1(C(CC2(C)CC2(F)Cl)=O)CC2(C1)SCCC2NC(C1CCCNS1(=O)=O)=O c1(C(N2CCCC(CN(C(=O)CCC(F)F)C)C2)=O)cc2n(c1)CCSC2 Cc1cc(S(=O)(=O)N(C)C(C)C)ccc1-c1ccnn1C(C)C c1(NC2CN(C(Cc3cn(CC)nc3)=O)CC23CC3)ncnc(CC)c1F C(=O)(CCCCC(C)=O)N1CC(CC(C(N2CCC(COC(C)=O)C2)=O)F)C1 c1(C(=O)NCC(CNC(C(CO)NC(C(C)C)=O)=O)O)cccc(Cl)c1O CN1C(=O)CN(C(=O)C(Cc2cn[nH]c2)NC(=O)C=CC2CC2)CC1=O c1(C(=O)NC(C2CC(O)CN2C(=O)OC(C)(C)C)C)cn(C)nc1C(F)F C1(C(=O)NCc2n(C)ncc2)C2CC1N(C(=O)CN1C(=O)CCCC1=O)C2 C(=O)(C(CCS(C)(=O)=O)n1cc(-c2cc[nH]n2)nn1)NCCOC(CC)(C)C C1(C(=O)N)CCN(Cc2cn[nH]c2)CC1.c1(N)cc(OCCO)ncn1 CCCCC(CCCC)C(=O)N(C)Cc1noc(C2CC2)n1 C1(C(=O)NC2CCCN(C(C3C(C)(C)C3C(F)F)=O)C2)CCC(C2CCC2)CC1 C(=O)(C(C)(C)C(=C)C)N1CCN(C(C(CC=C)NC(C)=O)=O)CC1 c1(C(=O)NC2C(CNC(=O)CCCn3cncn3)C2)cncc(F)c1Cl O=C1Cn2c(C(N3CC=CC3CNC(=O)CC3CCC(F)(F)C3)=O)nnc2S1 c1(C(=O)NC2(C(=O)NCC3CC3c3ccoc3)CC(O)C2)c[nH]c(=S)cn1 C1(NC(Cc2ccc(OC)cn2)=O)CCN(C(=O)COC(C)C)C12CCC2 CC1N(C(C2CC(C)N2C(=O)CC(C)(C)C#N)=O)CCCC1(C)C C1(CNC(=O)C2=COCC2)CC2COCC2N1C(c1coc(Br)n1)=O C12(NC(c3cc(Cl)c(Cl)[nH]3)=O)CCC(C1)N(C(C1CCCC1(F)F)=O)C2 C1(C(=O)Nc2c(C)cc(F)cn2)CCC(N)C(F)(F)CC1 N1(C(C(C)(C)OCC)=O)CCC2(C1)CN(C(=O)CSc1ccncc1)CC(C)O2 c1(C(=O)NC(C2(O)CN(C(C3CCOC3)=O)C2)C)cnc2ccnn2c1O C1(C(N(C)CC2(O)CCN(C(=O)C=C3CCCC3)CC2)=O)CCCCC12CCC2 N1(C(CC)=O)C2CCCC1CN(C(c1c(C)coc1C1CC1)=O)C2 C1(C(=O)NCC2C(CNC(c3cccnc3S)=O)C2)COc2ccccc2O1 C12(C(=O)NCC(C)OCCO)CC(CO1)N(C(C1(CC#N)CCCC1)=O)C2 Cc1c(CN2CC(O)CC2C(N2CCNC(=O)CC2)=O)ccc(Cl)c1F c1(CCNC(C2CC3CC3N2C(c2cccc(Cl)c2)=O)=O)ccc(Cl)cc1 N1(C(CCC(C)NC(Cc2c(C)scc2)=O)=O)CCC(N=[N+]=[N-])CC1 C1(C(N2CCC(NC(C3CCC(=C)CC3)=O)C2C)=O)OCC2CCCC12 N1(C(c2c(C)ocn2)=O)CCC(N(C(C2CCCN2C2CC2)=O)CC2CC2)CC1 N1(C(C2N(C(C)(C)C)CC2)=O)CC2CCN(C(=O)CC3(C#N)CCOCC3)CC12 Cc1ccc2occ(CC(=O)N(C(C)CCNC(=O)CN3CCC(C)C3)C)c2c1 C1(NC(C(C)=C2CC2)=O)COC2(CCN(C(c3cccc(C(C)Cl)c3)=O)CC2)C1 C1(CC(N2CCC(CN(C(=O)CN3CSCC3=O)C)C2)=O)CCCC(O)C1 CCCCCC(c1nnnn1CC1CCOC1)NCc1cncc(Br)c1 C1(C(N2CC(N(C)C(c3cnc(C(C)(C)C)o3)=O)C2)=O)Cc2c(F)cccc2O1 CC(C)(C)C(CC(=O)NOCC1CCCO1)NC(C1CCOC1(C)C)=O c1(C(N2CC(C(F)(F)F)CC(N)C2)=O)cc(F)cc(N=[N+]=[N-])c1 c1(OC)cc(C(N2CC(O)(CCNC(=O)Cc3ccnnc3O)C2)=O)ccc1F Cc1nn(C)c(C)c1CC(=O)NCC1COCCN(C(=O)C2=C(Cl)CCC2)C1 c1(C(N2CCC(C(=O)NCCOC)C2)C(=O)NCCC2CC2)cc(Cl)sc1Cl C(=O)(C(CC)CCCCC)NC1(CCNC(CSCC#C)=O)CCC1 N1(CCC)CCCC1C(=O)NCCn1ccc(C(=O)NC(C)C(C)F)c1 c1(C(=O)NC2(CN(C(=O)C(C(C)(C)C)C3CCC3)C)CC2)cccn2cncc12 N1(C(C2C(NC(CCSC(C)C)=O)CC2)=O)CC2CC(CN(C)C)C(C2)C1 c1(C(=O)N)cccc(Cl)c1.c1(C(=O)NC2C(CCOC)C2)sccc1CO C=CC(C)CC(=O)N1CC(OC)C(C(N2CCC2(CC)CC)=O)C1 N1(C(C(C)C(F)(F)F)=O)CCC2(CCN(C(=O)CSC(F)F)CC2)C1 C1(CC)CCCC(CNC(=NCCN2CCCC2)NC2CCCC2)CC1 C1(NC(c2n(COC)ncc2)=O)CN(C(c2cnn3c2OCC3)=O)CC(C)(C)C1 C(=O)(CC(c1ccccc1)C1CCCC1)NCCN(C)CC1(C(=O)NC)COC1 N1(C(C23CC(C#N)(C2)C3)=O)CC(C(=O)NC2CC(C(N)=O)C2)C2(CC2)C1 c1(C(C)C=O)ccc(C(N2CCC(C(C)NC(C3CC4CC4C3)=O)C2)=O)cc1 C1(C(=O)NC2C(NC(c3c(C(C)C)cccc3)=O)COCC2)CN(C)CC(C)O1 c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC2F)ccc2nc(OC)ccc2c1 C1(NCc2c(C)nn(C)c2Cl)CN(C(=O)CN2CCCCC2C)CCC1(F)F c1(CC)cc(C(=O)NC23CCC(C2)N(C(c2cnc(N(C)C)o2)=O)C3)ccc1Cl N1(C(C(C)n2ccnc2)=O)CC(C)C(C)(CNC(c2nnc(O)cc2O)=O)C1 c1(C(C)NC(=O)NC2CCN(c3ccc(C)cc3C)C2)cc2c(s1)CCCC2 N1(C(C)C(=O)N(C)C)CCCC(N(C(=O)CN(C)C(c2ccsc2)=O)C2CC2)C1C Cc1cc(CC(N2CCCC(NC(=O)C(C)C)CC2)=O)ccc1Br Cc1ccc(C(CNC(=O)C=CC(=O)N(C)C)NC(c2sccc2Cl)=O)cc1 c1(C(=O)NC(C2(O)CCN(C(C3(C)CCC3)=O)CC2)C)c2c(nn1C)CCSC2 Nc1ccc(CCC(N2CC(F)(F)C2)=O)nc1.C12CCCC(C1)C(=O)N2 N#Cc1cc2c(nc1N1CCCC(CNC(c3ccoc3Cl)=O)CC1)CCCC2 CCC(CC(=O)NC1CN(C(c2cccn2C)=O)C2(CCC2)C1)CC(F)(F)F C(c1ccccc1)=C(CC)C(=O)NCC(C1CC1)NC(C1CCCN1N=O)=O c1(OC)cccc(C(N2CC(NC(c3cn(CCO)nn3)=O)C(C)C2)=O)n1 c1(OCC(=O)OCc2c3nc(=N)[nH]n3ccc2)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NC(CCCC)CNC(C2(Cl)CC2)=O)cccc2c1OC(C)C(=O)N2 C(C)(C(C(=O)NCC1CN2CCC1C2)C(C)C)NC(c1c(C)ccnc1O)=O C1(COC)(CO)CCN(C(=O)NC(C2CCCO2)C)C1 CC1(C)CCC=C1C(=O)NCC1CN(C(=O)CCC2CCCC2)C2CC12 n1(C(C)C)ncc2cc(C(=O)NC3CC(CNC(=O)COC(F)F)C3)cnc12 C1(CC=C)(C(=O)NC(c2ccccc2O)C)CCCN1C(c1ccn(C)c1C)=O CCC(CNC(=O)C(=O)C(C)C)(CC)C(=O)Nc1conc1C c1(CNC2CC(C(N(CC(C)C)CC(=O)O)=O)C2)cc2cc[nH]c2cn1 n1(CC(N2C(CCNC(C3CN(C)C(=O)C3)=O)CCC2)=O)cccc(N)c1=O c1(C(=O)O)ccc(S(=O)(=O)NC2CC(C(=O)NCC3(O)COC3)C23CCC3)s1 c1(CC(N2C(NCO)CC2)=O)ccc(O)cc1.C1(OCCOC)CN(C=O)C1 c1(C(N2CC(NC(c3cn(CCCC)nn3)=O)(CO)C2)=O)c(OC)ccnc1F c1(COCP(C)(C)=O)csc(C#N)c1.C12CCN(C1)C(=O)NC2c1ccccc1 N1(C(C(CC)OCC)=O)CCCN(C(c2ccc(N)c(F)c2Br)=O)C(C)C1 c1(C(=O)NC(C)C(CO)NC(=O)Cn2ncnn2)ccccc1CC#N c1(C(N(CC(C)NC(C2(F)CC=CC2)=O)C)=O)cccc2cc(CCO)ccc12 CC1=NNC(=O)C1CC(=O)NCC=CCNC(=O)C(c1ccccc1C)(C)C CCC1=NOC(CC(=O)N(CCOCCCNC(=O)CC2COCC2O)CC)C1 c1(C(=O)NC(CCCC)CNC(C2CC2C2CCC2)=O)ccc2cc[nH]c2n1 C=CCCC(F)(F)C(=O)NC(c1ccc(C(C)C)cc1)CNC(=O)CCCCC C=CC(C)(CCOC)C(=O)NCCC(C)(C)NC(=O)C(C)C(O)CC C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(CC(=O)OC)C(c2ccccc2)C1 C=CC(C)(C)C(=O)NC1C=CC(CNC(C2CCC(=O)N2)=O)C1 CC1CCN(C(=O)CCN2CCCCC2=O)CC1CNC(c1ccno1)=O C=C(C)CC(C(=O)N1CCC(F)(C(=O)NC2(c3ccnn3C)CC2)C1)OC C1(CNC(C2(SCC)CC2)=O)CC(F)CN1C(=O)C=CC1CCCO1 C1(OC)CN(C(=O)C(C2OCCCO2)C)CC1NC(=O)Cc1ccccc1Cl c1(C(=O)NC2CCN(C(C3CCSCC3)=O)C2)cncc2c[nH]nc12 CCC(CCC(=O)NCC1(F)CCC(CNC(c2cn(C3CC3)cn2)=O)C1)OC C1(c2n(C(C)C)nnn2)(NC2(CF)COC2)CSC(C(C)C)C1 CC1CCCN(CCCCNC(=O)NCC(c2cccc(N)c2)O)C1 CCC(C(=O)NC1(C)CN(C(c2cccc(C(N)=O)c2N)=O)C1)C(C)O c1(CN(C(CC(COC)N)=O)C)cc(Br)cc2cccnc12 c1(COC(C2C(C(=O)NC3C(NC(CC=C=C)=O)C3)CC2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(C)N(C)C2CC2)cccnc1CO.c1(C(C(=O)N)O)ccccc1 C1(OC)CN(C(=O)CN2CCNC2=O)CCC1NC(=O)C(=Cc1cccnc1)C C1(NC(=O)C(C2CCC2)NC(c2nocc2Cl)=O)C2CCCC1CC2 C(=O)(CCCCCCC)N1C(C(=O)NC(C#CC)(C)C)CCC(C)C1 c1(C(=O)NC2CCN(C(N)=O)C(C3CC3)C2)csc2ccc(F)cc12 C(=O)(CC(C)(C)CN1CCOCC1)NC1C(CNC(CCCC#C)=O)C1 N1(c2snc(CC)n2)CCCC2(CC(NC(c3c(C)noc3C3CC3)=O)C2)C1 CCC(CC)CC(F)C(=O)N1C2CCC(C2)C1C(=O)NCCc1nccs1 CCC(CCC(=O)NCC1CN(C(c2[nH]nc(OC)c2Cl)=O)CC1O)OC Cc1nccc(C(=O)NC2CCCCC2NC(=O)C(O)CC(C)C)c1C CCCCCC(C)NC(=O)C=CC(C)NC(=O)C(CCC)N(C)C C1(NC(c2c(C)nc[nH]2)=O)CCN(C(=O)Cc2cc(Br)cs2)CC1C c1(NC(C2C3(CN(Cc4ccc(C)cc4Cl)C3)C2)=O)cnc2ccc(Br)cc2c1 N1(C(C2(C(N)=O)CC2)=O)CCC(NC(c2cscc2F)=O)C(CO)CC1 C(=O)(C1=CCS(=O)(=O)C1)NCC12C(CN(C(CCOCC#C)=O)C1)C2 N(C1c2ccccc2CC1(F)F)C(=O)NCc1ncn2ccccc12 c1(N(C)C)ccc(C(N2CCC(CCNC(C3(N(C)C)CCCC3)=O)C2)=O)cn1 c1(NC(=O)N2CCC2)cccc([N+](=O)[O-])c1.C1(C(C)C)(SC)CC1 c1(CNCC2C(C(=O)OC)CCC2)n[nH]c2c1CCCC2 Cc1ccc(C(=O)NCCC(O)CNC(c2ccc(C(C)(C)C)nc2)=O)cc1N c1(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)coc(=O)c2ccccc12 C1(C(C)C)C(=O)N1.N1(C(C(c2ccccc2)OCC)=O)CCC(SC)CC1 Cc1cc(=NCCC2CN(C)C2)[nH]c(N(C)CCc2ccc(F)cc2)n1 c1(C(=O)NCCN2CCN(C(c3occ(C)c3C)=O)CC2)ccsc1S(N)(=O)=O CC(C)CCC(O)C(=O)NCCC1CC(NC(=O)C=Cc2cccc(O)c2)C1 C(c1ccc(Cl)cc1F)=CC(=O)N(C1CCN(C(C(CC)OCC)=O)C1)CC C1(CNC(c2c(CC)ncnc2)=O)CC2CN(C(C3CCCCCCC3)=O)CC12 N1(C2CN(C(=O)NC(C)COCc3ccccc3)C2)CCCC1=O C1(NC(C(COCC)C)=O)CN(C(c2csc(CC(F)F)n2)=O)CC1O N1(C(CSCC(C)C)=O)CCN(C(=O)CC(C)CF)CC1CS(C)(=O)=O c1(CCC)noc2ncc(C(=O)NC(CC(=O)OC)C(C)(C)C)cc12 N1(C(CC2CC(NC(c3c(C)coc3)=O)C2)=O)CCC(F)(CF)CC1 N1(C(CCCn2cc(C(C(C)C)O)nn2)=O)Cc2ccccc2NC(=O)C1C c1(C(C2CCOCC2)C#C)nc(-c2ccc(C)cc2)nn1C1CCCC1 C1(C(N(CC(CC)CC)CC)=O)COCCN(C(c2cc(F)ccc2O)=O)C1 C(=O)(C#CC1CCCCO1)N(CC(CO)(CO)NC(C1CCCSC1)=O)C C12(C(N(CC(=O)OCC)CC)=O)CC1CN(C(=O)CCC1CCCC1)C2 c1(C(C)NC(c2ccc(F)o2)=O)ccc(CNC(c2cnc(O)[nH]2)=O)cc1 C(=O)(C#CC1(C)CC1)N1CCCC(N(CC#C)C(c2cnnc(C3CC3)c2)=O)C1 N1(C(C(C)SC(F)(F)F)=O)CCOCC1CNC(=O)C=CCOC1CCOCC1 N1(C(C=CC(=O)N(C)C)=O)CCCC1C1(O)CN(C(C2CC=CCO2)=O)C1 c1(CC(=O)NC2CN(C(C3(CC)CC3(F)F)=O)CC2F)ccc(C)c(O)c1 c1(C(N2C(CCC(=O)NCC=C(C)C)CCC2)=O)cc(C#N)ccc1N CS(=O)(=O)C1CN(C(c2c[nH]nc2CNC(C2CC(C)(O)C2)=O)=O)C1 C1(C(=O)NCC(CN(CC(=C)C)NC)O)CC2(C1)CC(C#N)C2 n1(CCOCC)nnnc1C(C1(C)COC1)NC(c1ccc(C)o1)C c1(OC)cnc(F)c(C(C(=O)NCC2CCCO2)N(C)CC2CCOC2)c1 C1(CNC(C2CC(OCC)C2)=O)CCCN1C(=O)C(Cc1ccsc1)NC=O C1(NC(c2c(OC)ccnc2F)=O)CN(C(=O)C(C)C2CCC2)CC(C)(C)C1 N1(C(C(CC)N(C)C)=O)CC2(CCC2)CC1CNC(C12CCOC1CCOC2)=O c1(CNC(C=C2CCC(C)C2)=O)cccc(SC)c1.C1(CC(=O)N)CCCSC1 N1(C(C(n2cc(Cl)cn2)C)=O)CCCC12CCN(C(=O)C(=O)NCC(F)F)C2 C1(O)(CC(N2C(C)CC2)=O)CCN(C(C2(F)CCOCC2)=O)CC1 CC1CCC(NC(c2coc(O)n2)=O)CN1C(=O)CN1CCCCCC1 c1(NC(CCC2N(C(=O)OC(C)(C)C)CCC2)=O)cc(Cl)c2n[nH]cc2c1 C1(C(N2CCCC(c3ccc(C)cc3)C2)=O)Cc2cc(F)cc(F)c2O1 N#Cc1c(F)cc(NC(=O)Cn2ncc3ncccc23)cc1Br NS(=O)(=O)c1ccc(O)c(C(N2CCOC(c3cn(C4CCC4)nn3)C2)=O)c1 n1(C(CC)C)ncc2cc(C(N3CCN(C(=O)CC(C)C)C(CO)C3)=O)cnc12 c1(CN(C)CCN)cn(CC(F)(F)CNC(c2ccsc2C(F)(F)F)=O)nn1 Cc1ccnc(C(=O)NC2CCN(C(C3CCC(=O)N3)=O)C2C(C)(C)C)c1 c1(CC(=O)N(C)CCc2cn(CC(=O)N(C)C)nn2)cn(C)nc1C(F)(F)F c1(C(=O)NC(CCCNC(C2CCCC(C(=O)OC)C2)=O)C)c(F)cccc1F C=C(C)c1ccccc1NC(=O)C(CC#CC)NC(c1cnc(NC)cn1)=O c1(C(N(C2CCCCC2)CCNC(CC2(C=C)CC2)=O)=O)c(C)coc1CSC c1(C(N(C2CN(C(CC)=O)CC23CC3)C)=O)c(F)ccc(O)c1F N1(C(CC(CC)CC)=O)CC(NC(C2C(F)(F)C23CC3)=O)CC12CCC2 C12(NC(c3c(C)snc3)=O)CCCCC1N(C(=O)CCc1cnc[nH]1)CC2 c1(C(COCC)(C)NC(C)C(C)C)nnnn1C1CCC1 C1(NC(CSCCOC)=O)CC(NC(c2cccc(F)c2N)=O)C12CCOCC2 C(=O)(CCCC(=O)NCC(O)CNC(C1CC2(CC(=O)N2)C1)=O)NC c12ccc(cc1)NC2CO.c1(CCCN)cn(CC(N2CC=CCC2)=O)nn1 CC1=C(C(=O)NCCOCC(=O)NCC2OCCCC2(C)C)CCO1 C#CC1CN(C(C23CCCCC2C3)=O)CCN1C(=O)CCOC1CCCC1 C1(NC(c2cocc2Br)=O)CN(C(C2CCCC2)=O)CC2(CC2)C1 CN1CCC(NC(=O)CC2(C)CC2)C12CCCN(C(=O)C1=CS(=O)CCC1)C2 c1(N2C3C(NC(C4CC(C)(F)C4)=O)(CCC3)CC2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(NC(C2OCC(=O)C2)=O)CN(C(=O)C(F)CC2CC2)CCC1C(F)(F)F N1(C(c2sc(C)c(Br)c2)C(=O)NCc2cccs2)CCC(CO)C(O)CC1 C(=O)(C(C1=NOC2CCCC12)N1CCCC(CC(C)C)C1)NC(C(=O)OC)C C12(NC(c3c(CC)scc3)=O)CCCCCC1N(C(=O)CC(=O)OC)CC2 C1(Nc2ncc(CC)s2)CCc2ccc(O)cc2C1.C12(F)CN(C1)C2=O c1(C(=O)NCC(N(C(CC(C(C)C)C)=O)C)C2CC2)cnn2cc(C#N)cnc12 N1(C(C)CNC(=O)C(F)CC2CCCCC2)CCN(c2ncns2)CC1 C(C)(C(=O)N1CC(C)(O)C1)(N(C)C(C1CN(C2CCCO2)C1)=O)C1CC1 Cn1[nH]c(=N)cc1C(=O)NCCC1CSCCN1C(=O)CC(=O)NCC1CC1 C(c1cccc(C)c1)=CC(N1CC(O)(C(C(=O)NC(CCC)CC)F)C1)=O N1(C(C(C(C)C)N(C)C)=O)CCC(NC(c2nn(C)cc2Cl)=O)C(F)C1 c1(C(=O)NCC2N(C(c3c(CC)noc3)=O)CC(O)C2)cc2sccc2n1C c1(C(C2C(NC(=O)NC(C3CCCN3CC(F)(F)F)=O)C2)=O)cccc(Br)c1 c1(OCC(=O)NC2CN(C(C3C(OC(C)=O)C3)=O)CC2C)ccc(F)c(Cl)c1 C1(C(=O)NC(CCCNC(C2(CC#C)CCC2)=O)C)CC(=C(F)F)C1 C12CN(CCN1)C2=O.C1(C)(C(=O)NC2C=CC(C(=O)OC)C2)CC(C)=NO1 C1(c2cn(CC)nc2)N(C(C(=O)NC(C)C(=O)OC)C(C)C2CC2)CC1(C)C N12CCC(C)C(C1)C(=O)NC(C)C2=O.CC1=CCN(C(=O)C2CC2)CC1 C1(NC(C(=O)N(C(c2ccc(F)c(F)c2)CO)C)=O)CCCC(C)(C)C1 c1(C(=O)OC)ccc(CC(=O)NCCOCCNC(=O)CCNSC(F)F)cc1 N1(C(C(C)N(C(c2cnc(OC)nc2)=O)CC)=O)CCCCC(C(=O)OC)C1 C(C(CC(C)C)C(=O)N1CCC(CO)(NC(=O)CC2(COC)CC2)CC1)OC C1(C(=O)NC(C2N(C(c3n(CC)nnc3)=O)CCC2)C)CCOC(CC)C1 N1(C(C(F)=C(C)C)=O)C2CCC(C2)C1CNC(c1nnn(C)c1N)=O CCC(C)(C)C(O)C(=O)NC(CNC(C1(CC)CCOCC1)=O)CC(F)(F)F c1(C(=O)NC2CCN(C(Cc3c(C)nc[nH]3)=O)C2)cc([N+](=O)[O-])c[nH]1 c1(C(N2C(CNC(CC(C)(F)F)=O)COCC2)=O)cccc(C(F)F)c1F Cc1cnccc1C=CC(=O)N(C)CCN(C)C(c1cocn1)=O N1(C(CSC)=O)CC2CCN(C(=O)CC34CCCC3C4)CC2C1 C1(NC(C(C)(C)c2ccc(Cl)s2)=O)CC(CNC(c2ccns2)=O)CC1O N1(C(C(C)NS(CC)(=O)=O)=O)CCCC2CN(C(C3CCCCN3N=O)=O)CC12 N1(C(c2cn3nc(C)sc3n2)=O)CCN(C(=O)CN2CC(C)C2)C(C)CC1C N1(C(=O)C#CC2CCC2)CC2CCN(C(c3c[nH]nc3C3CCOC3)=O)C2C1 CC1=C(C(=O)NC2CC(O)(CNC(c3cnn(C)c3C(C)C)=O)C2)CCO1 c1(NC(C2C(NC(c3cc(CC)no3)=O)CCCC2)=O)ccccc1N=[N+]=[N-] c1(OC)ccnc(CNC(=O)C(=O)Nc2ccnn2-c2ccc(Br)cc2)c1 N1(C(C(=O)Nc2cn(C)nc2)C2CC2Cl)CCCC2(CC1)CC2 CC1OCCN(C(=O)COC2(C)CN(C(=O)CCCn3cccc3)C2)C1C Cc1cc(C#N)cc(C)c1C(=O)NCC1(C)CCCN1C(=O)C=CC=C(Cl)Cl Cc1cc(NC(C2CC(C)N2C(c2ccnn2CCF)=O)=O)ccc1Cl c1(CC)onc(C(=O)NCc2cccc(C(N3CC(C#N)C3)=O)n2)c1C C1(C(N(C)CC2(CNC(C34CC(C#N)(C3)C4)=O)CC2)=O)CC2(CCC2)CO1 c1(C(C)Oc2ccccn2)cn(CCC2CN(C(C3(CO)CC3)=O)C2)nn1 c1(C(C(=O)NCCC(C)N(C(c2c(OC)csc2)=O)C)C)cccc([N+](=O)[O-])c1 C(=O)(C1=CCCOCC1)NCCCC1CCN(C(Cc2cc(C)no2)=O)CC1 C1(C(N(C(C)CNC)C(=O)CN(S(C)(=O)=O)C)=O)CC2(CCC2OC)C1 CC1=NOC(C(N2CCC(CCNC(=O)CN3CC(C)C3)C2)=O)C1C c1(C(=O)NCCC2N(C(CCCCC#C)=O)CC(OC)C2)cccc2c1OCC2 c1(C(N2CC(C)C(C)C2(C)C)C(=O)NCCCC)cc(OC)c(OC)cc1F Cc1cc(F)ccc1OCC1(N(C)C)CCOCC1 CC1C(=O)N(CC(N2CCC(CNC(N)=O)CC2)=O)C(=O)C1C.C1(C)(C)CN1 Cc1cc(=NCc2ccns2)[nH]cc1S(=O)(=O)NCC1CCn2ccnc2C1C c1(NCC(F)F)cc(=NCC2OCN2CC2(c3c(O)cccc3)CCC2)[nH]cn1 C(C(F)C(=O)NCc1ccccc1)C1CN(C(C(C2CC2)SC)=O)C1 C1(CNC(c2c(C)c[nH]c2)=O)C(C)CCCN1C(c1cc(CCO)on1)=O C1(NC(=O)CCc2ccsc2)CC2CC1CN(C(c1c[nH]nc1C(F)(F)F)=O)C2 c1(C(C(=O)N(CCNC(c2cccc(C)c2)=O)CC)C)ccccc1S(N)(=O)=O C12(C(=O)NCC3C4CN(C(C5CCCCS5)=O)CC43)CC3CC(CC(C3)O1)C2 C=CCCC(C)N=c1[nH]c(-c2c(F)cccc2Cl)cs1 C=C(F)C1(CC(=O)NC2(C3CCCN3C(C3(C#N)CC3(C)C)=O)CC2)CCC1 c1(C(N2CCN(C(c3c(C)nc(=N)[nH]c3)=O)CC2C)=O)cn(C)c(C)cc1=O Cc1cccc(Cl)c1CC=O.C1(NC(=O)COCCC(C)C)CN(CC)CCC1C CC1CCC(O)(CNC(=O)C=CCN(C)C(C2CC=CCO2)=O)C1 N1(C(C=CC=C(C)C)=O)CCCC(CNC(=O)CCN(C)C2CC2)CC1 CC(O)C(C(=O)N1CCCC(CO)C1)NC(=O)COCC(F)F c1(C(N2CCCC(CN(C(C(C)OC)=O)C)C2)=O)ccn2nccc2c1 CC1(C(=O)NCC(=O)NCc2cn(-c3ccccc3F)nn2)CCCC(F)(F)C1 c1(C(=O)NCC(CNC(=O)C(F)(F)CC2CC2)CO)c(F)ccc2c1OCO2 C(C)(C(C(=O)N(C(C)C(N)=O)C)C(C)C)NC(CCCOC(C)=O)=O c1(-n2c(C(n3cncn3)C)nc(-c3ccc(C)o3)n2)ccc2c(c1)OCCO2 N1(C(c2ccc(C)cn2)=O)CCN(Cc2ccc(Cl)c(C#N)c2)CC1C#N Cc1ccnn1C(C)C(=O)NC1CC1CNC(c1cc(CN2CCCC2)on1)=O c1(C(N(CC(CN(C(CCSC)=O)C)O)C)=O)c(Br)nc2n1CCOC2 C1(C(N(C)C)=O)CC(F)CN1C(=O)C(=O)NCC(F)(F)C1CCC1 c1(OC)cc(CC(=O)NC2(CCNC(C3CCNC3=O)=O)CC2)cc(F)c1 N1(c2cc(SC)ncn2)CCC2(CCCN2C(C2CCC(N(C)C)CC2)=O)CC1 CC1(C)CC(N=c2[nH]c3cccc(F)c3o2)CN(C(=O)COCCCN=[N+]=[N-])C1 C(C(C(=O)N1CCC1COC)NC(=O)C(C)=CCOC(C)=O)OCC Cc1cccc(C(=O)N(C2CCN(C(c3[nH]nnc3C(F)F)=O)CC2C)C)c1C CC1(C)CCC(C(N2CCC(CNC(=O)CC(C(F)F)n3cccn3)C2)=O)CC1 C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1CC(NC(Cc2c(C)nc(O)nc2O)=O)C1 c1(OC)cccc(CC(C)CC(=O)NC2(CN(C)C(c3ccco3)=O)CC2)c1 C1(CC)COC(C)CN1C(c1cccc(CNC(=O)C(C)(C)OC)c1)=O N1(C(C2(C(C)NC(CCc3ccc(C)o3)=O)CC2)=O)CCn2cnnc2C1 C(=O)(CC#N)N(CC(=O)NCC1(C)CCC1)CC#C c1(C(N2CCN(Cc3ccc(C(C)N(C)C)nc3)CC2)=O)cc(Br)ccc1I C1(CC(=O)NCC(C(=O)NC(c2csnn2)C)OC)CCC=CCC1 CCCC(CCC)CC(=O)NCC(CCC#N)C(=O)NCC1CCCN1C1CC1 C1(NC(c2ccsn2)=O)CC(F)(CNC(C2CCSC2)=O)C1 N1(C(c2c(C)coc2)=O)CCOC(CNC(=O)Cc2ccnc(F)c2)C1 C1(CC(=O)OCC2CN(c3ccccc3)C(=O)O2)CC2(CCOCC2)CO1 c1(OCC)ccsc1C(=O)NCC(C1CCOC1)NC(c1ccn(CCF)n1)=O C12(CNC(CC(C)O)=O)CCC1CN(C(c1ccc(OC3CCCC3)cc1)=O)C2 n1(CC(N2CC(NC(c3cc(-c4ccccc4)cs3)=O)(CO)C2)=O)cc(Cl)cn1 C(c1cnn(C)c1)=CC(=O)NC(CN(C(c1n(CC)nnc1)=O)C)C C#Cc1ccc(F)c(C(=O)NCC(C)N(C(=O)C(C(C)(C)C)SC)C)c1 C1(C(N2CC(CNC(c3cnc(OCC)nc3)=O)(CO)C2)=O)CC2CCC(C1)O2 Cc1c(C(=O)NCCCOC(C)C)ccn1OCCC(=O)NCc1nccn1C C1(OCCCNC(C2CC(O)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)CC1 c1(-c2scc(C(N3C(CC(=O)N4CCC4)CCC3)=O)n2)ccc(Cl)cc1F N1(C(c2nc(CC)sc2)=O)CC(NC(c2cc(C3CCOCC3)on2)=O)CC1C CC1C(NC(=O)CCCS(C)(=O)=O)C(C)CCN1C(=O)C1=CC2CCCC12 N1(C(C=C(C)C)=O)CCC2(CC1)C(N(C(=O)Cc1ccc(Cl)cc1)C)CS2(=O)=O C1(CNC(C2N(CCC)CCC2)=O)CCCCC1C(=O)NCC(=O)N(C)C CC(C)C(C(=O)NCC1CCCOC1)C(C)NC(c1cnnc(O)c1)=O CCCC1(C)C(=O)CNC(=O)Oc2cc(n(C)n2)C(=O)N1.C(C)(C)(C)OC(C)C c1(C(=O)NC2CC(C)(NC(C=CS(C)=O)=O)C2)ccc(=O)n(CC(F)(F)F)n1 c1(C(N(CCCCNC(C2CC(C)OC2)=O)C)=O)ccc(P(C)(C)=O)o1 N1(C(c2ccc(CC(C)C)s2)=O)CCC(C)N(C(c2ns[nH]c2=O)=O)CC1 c1(C(C(c2ccccc2Cl)F)Nc2ncc(C3CCCO3)s2)ccccc1Br Cc1nc(O)nc(C)c1C(=O)NCCN(C)C(c1cnn(C2CCOC2)n1)=O c1(C(=O)Nc2cc(C)c(Cl)nc2)ccc(S(C)=O)cc1 C=C(C)CCC(=O)N1CCC(O)(CNC(c2ccc(-c3cccc(Cl)c3)s2)=O)C1 C1(F)(C(=O)OCC)CN(C(=O)CC23COC(COC)(C2)C3)CC1c1ccccc1 c1(C(=O)NC2CCCC(CNC(=O)Cc3ccsn3)C2)ccn2nncc2c1 CC(C)CC(CNC(c1cc(CN(C)C)c[nH]1)=O)NC(c1ccccn1)=O C12(C(C)NC(C#C)C3CC3)CC3CC1C2C3 C1(CC)CC1(C1CC1)NC(=O)C(C)NC(=O)NCCC(=O)OCC Cc1cc(C(=O)N(C)CC2(O)CCN(C(=O)CCF)C2)cc(F)c1C c1(CC)c(C(=O)NC2CC(C)(NC(c3cccnc3S)=O)C2)cnn1C N1(c2cc(C(C)(C)C)ncn2)CCC2(CCCN(C(=O)Cn3ccnc3)C2)CC1 N1(C(Cc2nnc(C)o2)=O)CCN(C(C2CC2F)=O)C(CC(F)F)C1 C(C1Cc2ccccc21)c1n(C(CC)CC)nc(-c2ccccc2)n1 C1(C(C)C)CCC(C(=O)N(C2CCN(C(=O)CCF)C2)Cc2ccccc2)CC1 c1(NCCS(CC)(=O)=O)nc2ccccc2nc1NCC(c1ccccc1Cl)C S(=O)(=O)(c1[nH]c(=NC2CC(Cl)(Cl)C2)ccc1Br)N(C1CCCSC1)C c1(C(=O)NCCCC(C)(C)NC(C(CC)O)=O)nncc2c1CCCC2 c1(C(=O)OC)ccc(O)c(C(=O)ON2CC(CO)C3(CCC3)C2)c1 CC1=C(C(=O)N2CCC(NC(C3CCOC3c3nccn3C)=O)C(O)C2)CCC1 CN1CCN(C(C2C3CCCC3CN2C(C2CN3CCC2C3)=O)=O)C2CC12 N1(C(C2(O)CN(C(=O)OC(C)(C)C)C2)=O)CCC12CN(C(=O)C(F)CC1CC1)C2 C(=O)(C(C)(C)C1CCC1)NCC(=C1CN(C(C2(C(=O)NC)CC2)=O)C1)F C1(F)(CNC(C(C)CC2CCC2)=O)CCCN(C(=O)Cn2cc(Cl)cn2)CC1 c1(-c2cn(C(CNC(CC(C)C3CC3)=O)C)nn2)ccc(Cl)c(C#N)c1 Cc1cc(C)c(C(=O)NCC(C)NC(C23CC(C2)C(C)O3)=O)c(S)n1 C=CC1CCCCN1C(c1cc(Br)nn1C)C(=O)NCCCOC Cc1cc(CNC(=O)NC2COCC2(C)C)cc2c1CCC2 C1(C)(C(=O)NC(CNC(C#CC(OCC)OCC)=O)C(C)C)CCCCC1(F)F C(C)(C)(CN=c1cc(Cl)nc(C2CC2)[nH]1)NC(c1ccc2[nH]c(C)c(C)c2c1)=O CN1C(=O)CCCC1C(N1CCOCC1CC(=O)NCCC#CCO)=O c1(-c2sc(C(C)OC(=O)Cc3ccnc(O)c3)c(C)n2)ccccc1Cl C(=O)(CCCCCC(C)C)N1CCC(C(=O)NCc2c(C)occ2)C12CC2 c1(C(N2CC(F)(CNC(C3C(CC)OCC3)=O)C2)=O)cc2ccccn2n1 CC1(C)CCN(C(=O)C2=CCCCO2)C(C(=O)NCC(C)(F)F)C1 CC1=C(C(=O)N(CCN(C)C(C2CC3C=CC2O3)=O)C(C)C)C(C)(C)CCC1 C(=O)(CC(C)CC(C)(C)C)NC(CCC)C(=O)NCC(=O)NC1CC1 C1(C(=O)NCC2C(C(N(C)Cc3cc(OC)no3)=O)C2(C)C)CN2CCN1CC2 C1(C(N2CC(N(C(C3C(C)CC3)=O)C)C(C)(C)C2)=O)CN2CCCN1CC2 N1(C(C=C(C)Cl)=O)CCC(C2CCN(C(=O)Cc3ccnn3C(C)C)C2)C1 C(=O)(CCCC(N)=O)NC1CC(CNC(C(c2cn(C)nc2)(F)F)=O)CC1O N1(C(C2(C=C)CCCC2)=O)CCC2(CC1)CC2CNC(=O)CCC(C)(C)OC CCC(C)C(O)C(=O)NCc1csc(CNC(=O)Cc2cocn2)n1 C(=O)(C(Cc1ccccc1)NC(=O)CCCc1ccsc1)OCC#N n1(CC#C)cccc1C(=O)NC1CC(CC(=O)NCCCS(C)=O)C1 N1(C(c2scc(C)c2)=O)CCC2(CCCC2C(N2CCCC(C(N)=O)C2)=O)C1 N1(C(C2N(C(C(CCCC)C)=O)CCC(F)C2)=O)CCOC(C)(C)C1C C1(CC(=O)NC2(C(=O)N(CC3CCC3)CC3CC3)CCCCC2)CCCC1(F)F N1(C(Cc2c(C)ncs2)=O)CC(CNC(=O)CCNc2ccccc2)C(C)C1 C(=O)(C1CCCc2ccccc21)NC1C(NC(c2cc3oc(Br)cc3[nH]2)=O)C1 C1(CNC(c2c(C)occ2)=O)CCN(C(=O)C(c2cccc(CO)c2)=O)C1(C)C CC(CC(=O)N1CC(N2CCN(C(=O)CCCCCC#N)CC2)C1)C(F)(F)F C1(C(=O)NCC23CC2CN(C(C2CCCCN2C)=O)C3)(OCC)CCOCC1 CC(CS(C)(=O)=O)C(=O)NC1CC12CC(NC(=O)C(O)C(C)(C)C)C2 C(=O)(C1=NOC(CNC(C2(C#N)CCCC2)=O)C1)N(C1CCC(C)CC1)C Cc1cccc(Cl)c1C(=O)NC1COCC1NC(c1cncc(C)c1C)=O C1(NC(C(C)Cc2cnc[nH]2)=O)(CO)CCCN(C(C2CCOC2)=O)C1 O1NC(=N)CC(=O)OC(C)(N)c2csc(n2)C1.C1CCC1.CC N1(C(c2c(C)snc2)=O)CCN(C(=O)CN2CCCCC(O)C2=O)CC2(CC2)C1 c1(C(=O)NCC(CNC(c2ccnc(C3CC3)c2)=O)O)ccccc1-n1ccnc1 C#CC1(O)CC(C(N2CC(NC(=O)CC(O)c3ccccc3)C(CCC)C2)=O)C1 c1(C2N(C(c3nn(C)c(-c4ccc(O)cc4)c3)=O)C(C)CC2)c(Cl)cccc1Cl c1(C(=O)NCC(CC)NC(c2ccncc2Br)=O)c(C(C)C)nn(C)c1Cl c1(C(=O)NC2CCC(CNC(C(C(C)C)NS(C)(=O)=O)=O)C2)ccn(C)c(=O)c1 N=c1[nH]ccc(C(N2CCOCC2CCNC(=O)CC2C=CCC2)=O)c1Cl C1(CC(=O)NC2(CN(C(=O)C(=O)Nc3ccccc3)C)CC2)CCC(=O)NC1 c1(C(N2CCC(C(O)C3CC3)CC2)=O)ccnc(C2CC2)n1 N1(CC(=O)NC(C2(C)CC(=C)C2)=O)CC2CCC1C2.C(C)(C(C)O)N N1(C(C(CC(C)C)O)=O)CC2CCC1C(CNC(=O)C#CC1CCCO1)C2 C(=O)(C(F)C(F)(F)F)N1CC2C(CC(=O)Nc3cncc(C4CC4)c3)C2C1 c1(CC(NNC(=O)NC(C)Cc2ccnn2C)=O)ccc2c(c1)OCCO2 Cc1ccc(C(=O)NCC2CC3CN(Cc4cccc(F)c4F)CC23)n1C c1(CC)sccc1C(=O)NCC(C)N(C(=O)CCOCCOC)C C1(NC(CN2CCC(C)CC2)=O)C2CCC1N(C(=O)COC1CCC1)C2 N1(C(CC2CC(N(C)C)C2)=O)CC(F)CC1CNC(C1CC2(CCC2)C1)=O Nc1ccc(CN2CCCCC2Cn2cc(Oc3ccc(F)cc3)nn2)nc1 c1(C(=O)NC2CCC(NC(c3cn4ccsc4n3)=O)C2)cn2cccnc2n1 c1(C(N2C3CCC(NC(C=CC=CCC)=O)(C3)C2)=O)cnc2snc(C)c2c1 C(=O)(C(=O)NOC)NC(CCC)CNC(=O)CSCCC(C)C C12(C(=O)NCCn3cc(C(=O)NCC4CCCC4O)nc3)CCCC1C2(F)F N1(C(C2C(C#C)C2(C)C)=O)C2CCC(C2)C1CNC(=O)CS(=O)(=O)NC1CC1 CC1CN(C(=O)CCC2CCOC2)CCC1CNC(C1CCC(=O)O1)=O CC(C)C(F)C(=O)N1CC=CC1(C(=O)NCCCCF)COC C=CCC(C(=O)NC1COCC1NC(c1ncoc1C)=O)C(C)C C(=O)(C(C)(C(C)C)SC)NC1CC(CNC(Cc2cc(C(=O)OC)sc2)=O)C1 Cc1cc(C(=O)NCCCOCCCNC(C2(C#N)CCC2)=O)c(O)nn1 C1(C(N(CC(=C)C)CC(=C)C)=O)CN(C(C23CCC(CC2F)C3)=O)CC(C)O1 C1(C(=O)NC2(CC)CC2)CC(=O)N(CC(C)C)C1.C12(CCC1)C(=O)N(C)C2 C1(S(C)(=O)=O)(C(=O)NC2CCN(C(c3c(C)cc(CC)o3)=O)CC2F)CC(O)C1 CCC(CC(C)C)C(=O)N(CCCNC(C1C(Cl)(Cl)C12CC2)=O)C1CC1 N1(C(C2N(C(C)=O)CSC2)=O)CC=C(CNC(=O)C=Cc2ccnn2C)CC1 c1(OC)c(C(=O)NC2(CNC(C3(SC)CC3)=O)CCC2)ccnc1Cl N1(C(c2c(C(C)C)ccs2)=O)CCN(C(c2cccnc2OCCO)=O)CC(O)C1 C(C1OCc2cc(Cl)ccc21)NS(CC(CC)COC)(=O)=O C(C(C(=O)N1CCCCC1CN(C(=O)CC1(C)CCOCC1)C)C(F)(F)F)OC N1(C(C(C(C)(C)C)=O)=O)CCC2(CCC2NC(C2CCC(C)CC2)=O)CC1 C1(C(N2C(CC)CN(C(=O)CN3CCCCC3=O)CC2)=O)CC(C2CCCC2)C1 C1(CC)CN(C(C2CCC(=O)NC2)=O)CCC1NC(=O)C=Cc1ccccc1C N1(C(CCC(=C)Cl)=O)CCCC(C)(C)C1C(=O)NCCC(C)c1cn[nH]c1 C1(NC(C(C)NC(C2C3CCCC23)=O)=O)CCOC1CO.C(C)(C)(C)O Cn1cc(S(=O)(=O)NCC(=O)NCC(CO)NC(C23CC(CCO2)C3)=O)cn1 N1(C(CCN(CCCCOC)C)=O)CCC(C)(C)C1C(=O)NC1CCOCC1F c1(CC(C)C(=O)NC(C)(C)C(C)NC(=O)C=Cc2cscn2)ccc(F)cc1F c1(C(C(=O)NCC(=C)C)(C)N(C)Cc2sccc2C)cc(C)ccc1F c1(C(C)=O)cc([N+](=O)[O-])ccc1N1CC2C(C(N)=O)C2C1.N1CCCS1(=O)=O C1(NC(c2c(C)[nH]nc2Cl)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1O c1(C(=O)NCC2C(NC(C(CO)N(C)C)=O)COC2)ccc2cc(O)ccc2n1 c1(CC(=O)NC(CC)CN(C(c2nncn2C2CC2)=O)CC)cccc(F)c1F c1(C(N2C(C(N(C)Cc3cccc(C)n3)=O)C=CC2)=O)cc(C)c(O)nn1 Cn1cnc2c(NCC3(C4CCCCC4)CC3)nc(N3CCCC4(CC4)C3)nc12 n1(CC)ccc(=NC(=O)C23CC(CN2C(c2c(C)ccnc2O)=O)C3)[nH]1 CCC(CC(=O)N1CCCC(C)(CNC(c2nnsc2SC)=O)C1)C(C)C C(C(C(=O)NC1CC1OC(C)(C)COC)NC(=O)COC1CCOC1)OCC N1(CC)CCN(C(=O)C(C2CCC2)NC(C2CCCC2)=O)C(C)C1 c1(C(=O)NCCNC(c2c(CC(=O)OC)scc2)=O)nn(C)cc1Br C1(NC(=O)CC2(O)CCOCC2)CC2(C1)CC2C(=O)NC1CCS(=O)CC1 N#CC1(C(=O)NCC(C2CC2)NC(C2CC2C2CCC2)=O)CCOCC1 C1(CNC(c2ccc(C(N)=O)o2)=O)CN(C(C2CC=CC2)=O)C2CCCC2O1 N1(C(CCc2ccc(COC)[nH]2)=O)CCOCC(C(N2CC(=O)NC(=O)C2)=O)C1 N1(C(c2ccncn2)=O)CCC2C(CCN2C(c2c[nH]c(=O)c3ccnn23)=O)C1 C1(C(=O)NCC2(OC)CCN(C(=O)C#CC3CCC3)CC2)CCCC(C)(C)CC1 c1(C(=O)NCCCC(CCC)NC(=O)CCC(=O)NC)c2c(c[nH]c1=N)CCC2 C(CCCCC(=O)N1CCN(C(=O)C(F)n2ccnc2)CC1CF)N(C)C C1(C(=O)NCCc2cn(C3CCC(C)(C)C3)nn2)CCc2nn[nH]c2C1 c1(NCC2CC2)cc(O)nc(Cl)c1.c12ccccc1S2.C12CCCC(C1)NC2=O CN=c1[nH]cc(C(=O)NC(C)CCNC(=O)CCNC(=O)CC(C)C)o1 C1(C(=O)NCC2CCCN2C(N)=O)CCCC(C(N(CCCN2CCC2)C)=O)C1 c1(CN2CC3C(C(=O)NCCSC)(C3)C2)cc(C)ccc1C(F)(F)F CCC(C)CC(=O)C(=O)N1CCCCC1C(C)NC(=O)CCc1ccn(C)n1 c1(C(=O)NC(C(=O)NCC(c2nncn2C)C)Cc2cnc[nH]2)cc(Cl)n(C)n1 CC1CC(C(=O)NCCN(CC(F)F)C)N1C(C1CC(CCC(N)=O)C1)=O n1(C(C)C)cc(C(N2CC(C)(NC(=O)C3=CCSC3)C2)=O)c(Br)n1 CC1CN(C(C2CCN(C(=O)CC3CCCC(C#N)C3)CC2)=O)CC(=O)N1C c1(C(N2CCN(CCNC(c3ccccc3Cl)=O)CC2)=O)cncc(F)c1Cl c1(C(C)NC(=O)NCc2cc(CC)ncc2)ccc2nc(O)[nH]c2c1 CC1CC(=O)NC1C(=O)NCCC(C12CC3CC1C2C3)=O.N12CCC(CC1)C2 C1(NC(c2cn(C(C)C)nc2)=O)CC(O)CN(C(=O)Cn2ccc(C(F)F)n2)C1 C1(NC(c2cc(SC)oc2C)=O)CCCC12CCN(C(C1(C)C=CCC1)=O)CC2 C(=O)(C1=C(Cl)CCC1)NCC1(O)CC(NC(C(C(C)C)n2cncn2)=O)C1 N1(C(C2(C)C=CCC2)=O)CC2CCC1C(CNC(C1CCCN1C1CC1)=O)C2 CC(C)(C)C(CCO)NC(C1CCC2(CC2)N1C(=O)CCC(F)(F)F)=O c1(NC(CCC)C2CCC2)ncnc2c(C(C)C)nsc12 CC1CN(C(c2ccc(F)cc2)=O)CC1C(=O)NC1(C2CCCCO2)CC1 Cc1cc(Br)cc(C)c1CNC(c1ccc(Br)cc1Br)C CC(C)(C)C(C(=O)N1CCCC(CF)C1)NC(=O)COC1CC1 c1(OCCCC)ccc(CC(=O)NC(C)CCC2CCCC2)cc1OCC N1(C(c2ccc(C)[nH]2)=O)CC23CCCC2(C1)CN(C(c1c(Cl)csc1Cl)=O)C3 CCC(C)(C(=O)NC(CNC(=O)CCCCCc1cccs1)CO)C(N)=O CC(CNC(c1ccc(CNC(=O)OC(C)(C)C)cc1)=O)CC(F)F C12(CC)C3C4C1C1C2C3C41C.C12CCN(C1CO)C(=O)c1ccc(o1)C(=O)NC2 c1(C(=O)NCC2CC(CNC(C3C(C)(C(C)C)C3)=O)C2)cc(Cl)cn1C CC(C)(CC(=O)N1CCC(O)C1c1cccnc1)c1ccc(F)cc1 c1(COC(c2snc3cc(C(F)(F)F)ccc23)=O)ccc2cc(Br)ccc2c1 C(C(C(=O)NCC1(O)CCCC1)C(C)(C)C)NC(c1c(C)oc(C#N)c1)=O c1(CNC(=O)OC(C)(C)C)ccccc1COC(c1cocc1C(N)=O)=O C(=O)(CC(CN(C)C)C(F)(F)F)N(CC(C)N(C(C(CSC)C)=O)C)C c1(C(=O)NC(CNC(C(COC)O)=O)(C)C(C)C)[nH]cc2c1CCS2(=O)=O c1(C(=O)NCC(C(C)C)NC(C(C)SC(C)C)=O)ccc2ccnc(Cl)c2n1 Cc1nc(C#N)sc1C(=O)NC(C1CCCN(C(=O)CC(C)(C)C2CC2)C1)C N1(C(C2=CCC(NC(C(C(CC)C)N(C)C)=O)C2)=O)CC2(C1)OC(=O)NC2C C1(C)(C(N2CCC(NC(c3c(CC)n(C)nn3)=O)C2C)=O)CC(C2CC2)=NO1 CCC(C)(CCNC(=O)CC1(C)CC1)NC(=O)Cc1ccn(C)n1 c1(CNC(CCn2cc(C(CC)(O)CC)nn2)=O)cc2ncccc2cc1Cl N12CCC(C(C)C1)C2=O.C1(C(=O)OC)COCCC1NC(C)=O CC(C)C(C#N)C(=O)N1CC2CC2(NC(=O)COc2ccc(Cl)c(Cl)c2)C1 N1(C(C)=O)CCC2(CCCN(C(=O)C(F)OCOC3CCCCNC3=O)C2)CC1 N1(C(C2CC(C)(O)C2)=O)CCC2(CCCC2NC(c2ccc(CO)nc2)=O)C1 C1(NC(c2cc(NC(C)=O)ncc2)=O)CCN(C(=O)C(F)CC(C)C)C12CCC2 c1(C(=O)NC(CNC(C2(SC)CC2)=O)C)cc(N2CCC(O)CC2)ccn1 C1(NC(CCCCCC)=O)COC2(CCCN(C(c3ccc(F)cc3N)=O)C2)C1 C(=O)(C1=C(Cl)CCC1)N(CCNC(=O)CC1(C)CCOCC1)Cc1ccccc1 C(CC(C)C)(C(=O)N1CCC(C)(CNC(C2CCC(C)(F)CC2)=O)C1)OC C=C(C)CCC(=O)NCC1(CCOC)CCN(C(=O)C(C)OC2CCCC2)C1 C1(C(=O)NC(C)CC(=O)NCCSc2ccccc2)CCCCN1C(N)=O CCC(CCCC(=O)NCc1ccc(C)cc1F)NC(=O)Cc1cnoc1 N1(C(COCCCC)=O)CCC(O)(CCNC(c2cnc(OC)nc2)=O)C1 CC1CC(C)(C)N1C(C1CCN(C(=O)CCc2ncccn2)C1)=O C(C(=O)NCCC1CC1)(C1=CCSC1)N(CC(C1CCOC1)C)C C1(CNC(CN(C(C)=O)C)=O)CCN(C(c2ccc(-c3cccs3)[nH]2)=O)CC1 c1(C(=O)NCC(C2CCCC2)NC(C(CC=C)(F)F)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(=O)CSC(F)F)CCC(Nc2nccc(CO)n2)CC1 C(=O)(CC(C)(C)OC)NCCC1(OC)CN(C(=O)CCOCC(F)(F)F)C1 c1(C(=O)NCCOCCN(C(=O)CC2CC(F)C2)C)ccc2ccccc2c1 C1(NC(C2(OC)CCOC2)=O)CCCC(NC(=O)Cc2cscn2)C1 C(CCNC(=O)COCc1cn(Cc2ocnc2C(=O)O)nn1)(C(F)(F)F)OC CC1C(NC(c2cncc(CO)c2)=O)CCCN1C(c1ns[nH]c1=O)=O c1(CC(=O)NC(CNC(C(CC)C(F)(F)F)=O)C2CC2)c(C)oc2ccccc12 C1(C(=O)NCC#CCCO)(OC)CCN(C(=O)CC2CCCCO2)C1 C(C1CN(C(=O)CCn2ccnc2)Cc2ccccc21)NC(=O)Cc1ccco1 N1(C(C(C)n2cccn2)=O)C2CCCC1CN(C(=O)C1=NOC3COCC13)C2 C1(C(=O)NC2(CCCC)CC2)CN(C)CCN1C(=O)CCCCOC C1(NC(c2ccc(SC)o2)=O)CC(NC(c2ccnnc2O)=O)C12CCOCC2 CCC(C(=O)NC1(C)CN(C(=O)C(=O)NC2CNC(=O)N2)C1)Oc1ccccc1 C(=O)(CC1=CCOCC1)NCC1CCN1C(C1CCCCC1c1nc[nH]n1)=O C(C(C)(C)C(=O)NC1CCCC1CC(N1CC(NC(N)=O)C1)=O)SC N1(C(C2C(C)OC(C)C2)=O)CCC2(CCC2)C(CNC(c2ccncc2O)=O)C1 c1(C(N2CC(CNC(C(C)OC)=O)C2)=O)cc(C)oc1C(F)(F)F C(CCC(C(=O)N(CC(C)C#N)C)NC(c1ccc(CO)o1)=O)OC S(=O)(=O)(c1ccc2c(c1)NC(=O)CCS2)N1CC(C)N(C)C(C)CC1 c1(C(=O)NC2C(NC(=O)C(O)Cn3cncn3)C2)cncc(F)c1 N1(C(CC2CCC(=O)N2)=O)CC2CCN(C(c3scnc3Cl)=O)CC2C1 CCCC(C)(O)C(=O)NCCCOCCC(=O)NCCCCC1CCCC1 C12(NC(=O)C=C(Cl)Cl)CCC(CC1)N(C(C1CC1c1cccc(F)c1)=O)C2 C1(C)(C(N(C2CCCN(C(CN(S(C)(=O)=O)C)=O)C2)CCF)=O)CCS(=O)(=O)CC1 N1(C(C(C(C)C)(C)O)=O)CC2CC(O)C1C2NC(c1cc(C(F)(F)F)nn1C)=O c1(CCC(=O)NC(CNC(=O)C=Cc2cscn2)CO)cnc2ncccn12 C12(C(=O)NCCC3OCCN(C(C4CC5CC5C4)=O)C3)CCC(CC1)CC2 CCCC(C(=O)N1CCCC1CN(C)C(C1C(C)C1C)=O)OCC Cc1nc(C)c(C(=O)N(C)CC2(O)CN(C(=O)CCC3CCCN3C)C2)o1 N1(CC(C)S(C)(=O)=O)C(=O)CCN(CCC23CCC(CC2)OC3)C1=O C1(CNC(=O)Nc2sc(Br)c(C)c2C)CC2(C1)C(F)(F)C21CC1 C1(NC(=O)C=CBr)COC2(CCN(C(=O)Cc3cnc4ncccn34)CC2)C1 C1(CNC(C)=O)C(C)CCN1C(c1cnc(Cc2cc(C(F)F)cs2)nc1)=O C(=O)(CCC(=O)NC1CCOCC1C(=O)NC(c1ncco1)C)NCC C(C(C)(CC(C)C)NC(c1cc(Cl)c[nH]1)=O)NC(c1cnn(C(CC)C)c1C)=O C1(C(=O)NCCN2CCCNC2=O)CC2(CC2)CN1C(C1CC2C=CC1C2)=O Cc1ccc([N+](=O)[O-])cc1C(=O)NC(C)CCNC(C1(S(N)(=O)=O)CCCC1)=O S(=O)(=O)(c1cccc(C(=O)O)c1)N1CC(C)(C(=O)Nc2cc3cnccc3[nH]2)C1 c1(CC)cc(C(N2CC(NC(=O)CCS(N)(=O)=O)CC(C)C2)=O)cc(O)n1 C1(C(=O)NCC(C(C)C)NC(C(CC)n2nccc2C)=O)CCC(C2CC2)CC1 Cc1cc(C(=O)NC2CC(C)N(C(=O)CSc3nncs3)C2)cc(C)n1 C1(C2C(CN3CC(C4OCCN(C(C(C=C)C)=O)C4)C3)C2)CC(C2CCCC2)C1 C(=O)(C(C(C)(C)C)NC(N)=O)N(CC(O)CNC(c1[nH]ccc1C1CC1)=O)C N1(C(C(CCC#C)NC(=O)C(C#N)CC)=O)CC2CC(F)CC2C1 CC(C)C(CN(C)C)C(=O)N1CCCC(CNC(c2ccnnc2O)=O)CC1 CN=C(NCc1ccc2cc(C)[nH]c2c1)N1CCC(CC)C1 Cc1cc2[nH]c(C(N3CCC(O)(CCNC(c4cnc(O)o4)=O)CC3)=O)cc2s1 C(CCC(C)(C)NC(=O)CCC1CCC(C)O1)NC(C1(CC=C)COC1)=O N1(CC(=O)NCC(C2CCCCC2)NC(C=CCC)=O)CCP(C)(=O)CC1 C1(CC(=O)NC(C(=O)OC)CO)CCCCN1C(=O)CC1CCCC(=O)C1 c1(OCC(=O)N(CCC(Cl)Cl)CCN(C)C)ccc(Cl)c(F)c1 C1(C(N2CC(N(CC=C)C)C2)=O)(NC(=O)CCSCC)CCCC1C C(=O)(C1c2ccccc2OCC1(C)C)NC(CN(C(C1(C)CC(=C)C1)=O)C)CC C1(C(=O)NC2C(C(=O)NC(C(=O)NCC)C)CC2)CC2(CCC2)CO1 CC(C)CCC(=O)NCC(=O)NCC1CCCCC1N(C(C12CCC1CC2)=O)C1CC1 C(=O)(C(C(=O)N1CCC(N(C)C(c2coc(C)c2)=O)C1)c1ccccc1)OCC N1(C(C(c2ccccc2F)(C)C)=O)CC2C(NC(C3CN(C4CCC4)C3)=O)C2C1 c1(NC(c2scc(C(=O)Nc3cc(O)n[nH]3)n2)=O)ccc2[nH]c(=O)ccc2c1 c1(CCC)ccc(NC(C2C(C)CCN2C(=O)C=CCO)=O)cc1 c1(C(N(CCOCCCN(C(CC(CC)C)=O)C)C)=O)cnn2c1OCC2 C1(C(=O)NC(C2CCCN2C(C2CS(=O)(=O)C2)=O)C)CCC(=O)N1C C1(NC(C(C)=C(CC)C)=O)CC(NC(=O)Cn2nc(C)c(Cl)c2C)C12CCC2 CC(C)(C)C(CNC(=O)CC1CCC(=O)CC1)C(=O)NCCOCC1CCC1 C1(NC(c2cc(OCC)ncc2)=O)CN(C(C2CC2C2CCCO2)=O)CCC1C O=C1CS(=O)(=O)CC(C(=O)NC2CCN(C(c3ccc(O)nn3)=O)CC2CO)N1 C1(N(CC#C)C(c2ccoc2)=O)CCN(C(=O)C(C(=O)OC)OC)CC1 c1(C(=O)NCC)c(F)cccc1F.N12CCC(C1)N(CC)C(=O)C2 c1(OC)cc([N+](=O)[O-])ccc1C(N1CCN(C(=O)CNC(N)=O)CC1C(F)F)=O c1(C(N2CCC3(CC3C(=O)N(CCO)CCO)C2)=O)ccc2n[nH]cc2c1 C(N=c1[nH]c2c(c(=NCCC(C)(C)C)[nH]1)CSC2)C1(COC(C)C)CCOCC1 c1(CSc2c(-c3nc(N4CCCC(C)C4)sc3)cccc2)n[nH]c2c1COCC2 Cc1c(Cl)ccnc1C(=O)NC1CCCC(NC(=O)C2=C(Cl)CCC2)CC1 c1(C(=O)NCCCNC(C2(C)ON=C(C)C2)=O)ccc2c(c1)CCC(C)N2 C1(C(N2CC(C)C(NC(=O)CCOC3CCCC3)C2)=O)COc2ccccc2C1 C1(C(N2CCN(CC)CC2C)=O)CCN(C(=O)CCNC(=O)COC)C(C)(C)C1 c1(NC(C2(CN)CC2)=O)cc(Cl)cnc1Br.c12ccc(cn1)[nH]c2=O C1(OC)CCCCC1C(=O)NCc1cccc(Nc2ccnn2C)c1.C(N)(=O)NC c1(OC(C)C)ccccc1C(=O)NNC(=O)N1CCC1C1CCOC1 C1(C(=O)NC2CC(CNC(C3(C)CCN(C)C3=O)=O)C2)CCC(F)(F)CC1(C)C C1(C)(COC)CC(NC(c2cscn2)=O)CN1C(c1c[nH]c(=N)s1)=O C(c1ccc(F)c(F)c1)=C1C(C(=O)NC(CCC#N)C(N)=O)CCCC1 C#CCC(C)(CC)C(=O)NCCOC1CCN(C(C2(C)CCCCO2)=O)C1 N1(C(C2(C)CCC2)=O)CCN(C(c2cn(CC(F)F)cn2)=O)C2(CC2)C1 C(=O)(C(C)(C)Cc1ccccc1Br)N(C(C)COC)CC=C CC12CC(NC(=O)C#CC3CCCOC3)(C1)C1(CCN(C(=O)COCCF)CC1)O2 N1(C(C(C(C)C)O)=O)CC(NC(C2CC(OC(F)(F)F)C2)=O)C2CCCCC12 c1(C(N2CCC(CNC(C(CC#C)C3CC3)=O)(OC)C2)=O)ncnc(C)c1C Cc1csc(CN(C)C(c2c[nH]nc2CCNC(=O)C(C)n2cncn2)=O)n1 C1(CC)CN(C(=O)CN2CC(C)(OC)C2)CCN1C(=O)C(N1CCCC1)C1CC1 Cc1c(F)ccc(Cl)c1C(=O)NCC(C)(C)NC(=O)CC(C)C1CCCO1 CC(C)(C)C1=NOC(C(=O)NC2CCCCC2CNC(=O)CSC2CC2)C1 Cc1c(C(N2CCCC(C(=O)NCCCP(C)(C)=O)CC2)=O)c[nH]c1C#N S(=O)(=O)(c1ccccc1Br)N1CCN(C(=O)Nc2ccc(C)c(Br)c2)C(C)C1 Cc1cc(C(=O)NC2COCC2NC(c2cnc(C(N)=O)s2)=O)c(C)c(C)c1 c1(C(=O)NCC(CNC(=O)C(C2CCCC2)OC)OC)c(F)ccc(O)c1F c1(CC(=O)NC23CC2CN(C(c2scnc2Cl)=O)C3)ccc(F)cc1F c1(NC(c2nnco2)C)nc2ccccc2cc1Cl N1(C(=O)CC2CS(=O)(=O)CCO2)CCc2cc(C3CC3)ccc2C1 c1(OC)cc(Cl)ccc1C(=O)NC1CCCC(NC(C2(C)C=CCC2)=O)C1 C(=O)(C1OCCn2ccnc21)NC1CC(CCNC(=O)CCc2cnn[nH]2)C1 Cc1ccc(C)c(C(=O)NCC2CCN(C(c3cccc(CS(C)=O)c3)=O)C2)n1 C(=O)(CCCCCCC)N1C(CC(=O)N(C(C(=O)NC)C)C)CC(C)(C)C1 Cc1[nH]nc2c(C(N3CCCC(C)(C)C3CNC(=O)CO)=O)cccc12 N1(C(COCC=C)=O)CC2C(C(=O)NC(C)CCC3CCCO3)C2C1 CC1OCCC1(F)C(=O)NCc1nocc1C(=O)NC1CCN(C2CC2)C1 CN=c1[nH]cc(C(N2CC(NC(c3cc(C(F)F)nn3C)=O)C3CC23)=O)s1 C1(C(=O)NC(C(N2CC(C)SCC2)=O)CO)C2CCC(C2)C1C Cc1nc2c(o1)CCN(C(=O)C(=O)NCC1(C)CC(N)C1)C2 N1(C(c2nn(C)c(Cl)c2)=O)C2CCC1CC(NC(c1cncn1C1CC1)=O)C2 C(C(F)(C(=O)N1CCCC1C1CCOC1)C(C)C)NC(c1ncn(CC)n1)=O C1(C2(O)CCN(C(=O)C(C#N)CC)CC2)(NC(C=CC=CCOC)=O)CC1 N1(C(c2cnc(CC)o2)=O)CCCC2C1CCCN2C(C1CCC=CCCC1)=O C1(OCCNC(c2c(CC)c[nH]n2)=O)CCN(C(=O)COC(C)=O)CC1 C1(CC)(NC(C2CCCOCC2)=O)CCCN(C(c2oc(C)cc2C)=O)C1 c1(C(N2CC3C(CNC(c4c(OCC)cccc4)=O)(C3)C2)=O)cc(C)ccc1I C1(C#N)(C(=O)NCCCCc2cn(-c3ccc(C)cn3)nn2)CC12CCC2 c1(C(=O)NC(CN(C(C(CC)(C)C#N)=O)C)C)ccc2nc(C)oc2c1 CCC(C)CCC(=O)NCC(CNC(=O)CSCc1csc(C)n1)OC c1(C(=O)NC2C(SC)CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)ccn2c1CCCC2 c1(NC(Cc2ncc(-c3ccc(OCC)nc3)cn2)=O)cc(Cl)cc(Cl)n1 C1(C(=O)NC2CCN(C(COCCCC)=O)C2)CCN(c2cccc(Cl)c2)C1=O N1(C(C=CCNC(c2c(CC)c[nH]c2)=O)=O)CCC(O)(CC)C1 C1(C(N(C2CCCN(C(C3(C)CCCC3)=O)C2)C)=O)CCN(S(=O)(=O)N(C)C)C1 N1(C(COCCOCC#C)=O)CC(O)(C(F)C(N2CC(CN(C)C)C2)=O)C1 c1(C(N(C)CCNC(C2CC(C)(F)C2)=O)=O)c[nH]c2cccc(F)c12 C=CCC(C(=O)N(C1CC1)Cc1cn(CC2CC3CC3C2)nn1)NC(C)=O Cc1cccc(OCC(=O)NCCCN(C(C2CC(C)CCO2)=O)C(C)C)c1F C1(NC(C(CCCC)O)=O)CCCCN(C(c2cncc(C3CC3)c2)=O)CC1 c1(NC(C2CCC(CNC(C(C=C)OC)=O)C2)=O)cnc2ncnn2c1 c1(C(=O)NCC23C(CN(C(C4CC(C(C)(C)C)C4)=O)C2)C3)cnc2nccn2c1 c1(C(N2CC3CN(Cc4ccc(F)cn4)CC3C2)=O)c[nH]c2nccc-2c1 c1(C(=O)O)cc2ccc(Cl)cc2nn1.c1(OC)cnc(CN2CCN(C(C)=O)CC2)cn1 c1(C(N2CCC(CC3CC3)C2)C(=O)NCC(F)F)cn2c(Br)cnc2s1 c1(COC)ncc(C(=O)NC2CCCCC2NC(C2CCCCC2C)=O)c(O)n1 c1(C(C)(C)CC2CCC(Cc3nc(C(F)F)no3)CC2)ccc2ncccc2c1 c1(-c2nc(-c3cccc(OC)c3)nn2C2CC2C)cc(Cl)nnc1O c1(OC)cc(C)nc(O)c1CN(CCNC(=O)Cc1c(C)cccc1Cl)C1CC1 n1(C(C)C)cc2ncc(C(=O)NC3CCN(C(=O)Cc4cc[nH]c4)CC3O)cc2n1 C=CC1(CO)CCN(C(=O)CC(=O)OCC2CCn3ncnc3C2)CC1 c1(CC)nonc1C(=O)NCCCCC1CN(C(=O)C(C2CC2)C2CC2)C1 CCN=C(NCC1=CCCC1)N1CCC(c2cc(F)c(F)c(F)c2)C1 C1(NC(C(CNC(=O)CSc2nc[nH]n2)OC)=O)CC2(CCCCC2)C1 C1(C(=O)NC2C(CNC(=O)CCCn3cncn3)C2)CCCC12CCC2 C1(C2CC2)(CNC(c2c(CCC)nco2)=O)CCN(C(=O)CCCC#N)C1 C1(CC)(NC(C2CC3(CC3)C2)=O)CCCN(C(=O)CNC(C)=O)C1 C(CC(C(C)(C)C)NC(C1CCCS1)=O)N(C)C(C1CCC=CCC1)=O CS(=O)(=O)C1CC(C(=O)NCC2CC(NC(=O)Cc3cc[nH]n3)C2)C1 N1(C(C(F)=CC)=O)CCCC2(CCN(C(C)C(=O)NC(C)CC)C2)C1 c1(NC(C2C(C(=O)OC)C2)=O)cc(C(=O)Nc2cc(I)ccc2C)cc(Cl)c1 C(CC(C)(C)NC(=O)Cc1ccsn1)=CC(=O)NC(C1CCC1)C c1(CN2CCC(SC(CC=C)Cc3nccn3C)C2)oc(SC)nc1C N1(C(C(C)(C)F)=O)CCC(C2CCCN(C(C3CC(=O)NC(=O)C3)=O)C2)C1 C(c1ccc(C)cc1)=CC(=O)NC(CNC(c1oc(CC)c(C)c1)=O)CCOC Cc1c(Br)ccnc1C(=O)NC1CC(CO)N(C(=O)C(F)CC2CC2)C1 c1(C(N(CC(C)N(C(C2(COC)CCCO2)=O)C)C)=O)ccc(C2(C)CC2)cc1 N1(C(CC=C)=O)CC2CCN(C(c3cc(N4CCCC4)ccn3)=O)C2C1 c1(C(=O)NCCC2(OC)CN(C(=O)CC3CCC(=O)N3C)C2)ncn2c1CCC2 Cc1cccc(C)c1C(CO)NC(=O)C(F)(F)C(O)C1CC1 c1(OCCC)cc(F)ccc1CNC1CCC(C(=O)N(CC(C)C)CCO)C1 N1(C(C(C)N(CC)CC)=O)CCCCC(C2CN(C(C3(C)CC3C)=O)C2)C1 CC(CCC1CC1)NC(=O)CC=CCNC(=O)CC1CSCCO1 C1(CC(=O)NCCC#C)COC(C)(C)CN1C(=O)COCCCC(C)C Cc1cnn(CCC(=O)N(CCC(c2ccc(C(=O)OC)[nH]2)=O)C)c1.C(CCN)O Cc1ccc(C(C)C(N2CCC(N(C(=O)CN3CCCOC3=O)C)CC2)=O)cc1 CC1CCCC(CC(=O)NC(C)CN(C)C(C2CCCC(=O)N2)=O)C1 c1(CC(=O)NC(C2CCCC2)CNC(CN(CCC)C)=O)c(C)cc(C)nc1O C1(N(C(C=C(CC)CC)=O)CC)CCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)C1 c1(C(=O)NCC(CC)NC(C2CCC(OC)C2)=O)sc(S(N)(=O)=O)cc1C C1(N(C)C)CCC(C(=O)NCCCCNC(=O)CO)C1 c1(OC)ccc(F)cc1C(N1CC(NC(c2cc(C)ccc2Cl)=O)CC1C)=O CC(C)(C(=O)NCC1CC2CCC1N2C(C1CCCC(=O)O1)=O)C(F)(F)F Cc1ccccc1C(C)C(=O)NCCC1CCCN1C(C1CCC1C(C)(C)C)=O c1(CC(=O)OC)[nH]ccc1C(=O)NC1CC(N(C)C(c2cc(C3CC3)on2)=O)C1 Cc1cccc(Br)c1C(CNC(C1COCC(C)(C)O1)=O)NC(=O)CO CCCCC(CC)C(=O)NC(C(=O)NCC1CC2CCC(C1)C2)C(C)(C)C CCC(O)C(F)(F)C(=O)NCCC1CCCN1C(C12CCCC1CCC2)=O C12(C(N3CC(CC)C(NC(C4(CCN(C)C)CC4)=O)C3)=O)CCC(F)(CC1)CC2 Cc1nnc(O)c(C(N2CC3CC3(CNC(C3CN(CC(C)C)C3)=O)C2)=O)c1C c1(C(=O)NCC2CC(NC(C(CC)(F)F)=O)C2)cc(C2(C)CC2)ccc1F C1(C(=O)OC)CC12CN(C(=O)C(C)(O)CC(=O)NC1CC1CC(C)(C)C)C2 C=CCCC(C(=O)NCc1cc(C(N)=O)co1)NC(=O)C(F)C1CC1 N1(C(c2c(CC)nsc2N)=O)CC(c2cc(C)[nH]n2)C(C)(C)C1 C(=O)(C(O)C1CC1)N(CCOC)CC1CCCO1 c1(N2CCCC(OC)(CN(C)C)C2)cc(Br)ccc1S(=O)(=O)NC1(C)CCC1 c1(C(=O)NCC(C)NC(CC(CCC)C)=O)cc(Cl)c2ccccc2c1O c1(C(=O)NCCN(C(C=C(C)c2ccccc2)=O)C)ccc2c(c1)N(C)C(=O)C2 c1(C(=O)NCC(C(C)C)NC(=O)Cn2cc(Cl)cn2)ccc2ncnc(O)c2c1 C(C(CNC(c1ccccc1C(F)F)=O)C(F)(F)F)NC(C=C1CCN(C)C1)=O N1(C(Cc2cccc(CC)c2)=O)CC(F)(F)CC1(C)CNC(c1cc(C)co1)=O C#Cc1ccc(C(N2CC3(CC3)CC2C(N2CC3CC2CN3C)=O)=O)c(Cl)c1 C1(CNC(CS(CC)=O)=O)CCN(C(c2cccc(N3CCCC3)n2)=O)C1(C)C CC(C)CC(C)(CNC(C1(C)CC2CC2C1)=O)NC(C1CCC2(CC1)CC2)=O CCC(C)(CC)C(=O)N1CCC(C(=O)N(C(C)C(=O)NC)C)CC1 c1(CC(C)N(C(C(=O)NC(N)=O)C(C)C2CC2)C)ccc(F)c(F)c1 C1(C(C)NC2CCN(C(=O)CC3CC3)CC2)CCCCN1C(=O)COCCCF C1(N(C(c2c(C(C)(F)F)cccc2)=O)CCO)CCN(C(=O)C=C2CC2)CC(O)C1 C1(NC(CN(C(C)=O)C)=O)CN(C(=O)C(C)NC(N)=O)CCC1O Cn1c(C(=O)NCC(C(C)(C)C)NC(C2(CO)CCCC2)=O)cnc1O CC1(C)CC(C)(CNC(c2cnsc2)=O)CN1C(=O)CC1CCCO1 C1(NC(C(C)CSC(F)(F)F)=O)CCCCC1NC(c1ccc(C(F)F)nc1)=O N1(C(C(C)OC2COC2)=O)CC2(C1)CN(C(C1CC1c1cnc[nH]1)=O)CC2CO N1(C(C2CC(NC(c3cc(OC)cc(Br)c3)=O)C2)=O)CCc2ncccc2C1 C(=O)(C(F)(F)CC(C)C)N(CCC)CCNC(c1nccc(Cl)c1Cl)=O N1(C(c2cscc2C)C(=O)NC(CC)(C)C)CCCC(CNC(C)=O)C1 c1(C(N2C(C(N3C(C(=O)OC)CC3)=O)C=CC2)=O)cccc(=O)n1C CC(C)C(C(=O)N1CCC=C(F)C1)C(C)NC(=O)CN1CC2CC2C1 c1(OCC=C)ccc(Cl)nc1C(=O)NCC1CCN(C(=O)CCC#N)C1 C(=O)(C(O)C1=CCCCC1)NC1C(n2cc(C3CC(C(=O)O)C3)nn2)CC1 C1(CC(=O)N(CC(C)NC(c2c(CC)onc2)=O)C)CCCNC(=O)C1 C(=O)(NN1CCCC1C(N1CC(COC(C)=O)C1)=O)c1c(CC)nccc1 Cc1cc(C(=O)NCC2(NC(=O)C(c3cccc(F)c3)F)CCOCC2)[nH]c1C c1(C(N2CCCN(C(c3cn(C(C)C)nn3)C)CC2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N2CCCC(N(C(C3N(C(C)C)CCC3)=O)C)C2)=O)cc2c(ccn2C)s1 O=S(=O)(c1c[nH]ccc1=Nc1ccncn1)N1CCS(=O)(=NC=O)CC1.C1CC1 N1(C(c2c(CC)nns2)=O)CC2COCCC2(NC(=O)CCN2CCC2)C1 N1(C(COCC)=O)CC(NC(=O)C2=CCCC2)CC2(CCOCC2)C1 c1(C(=O)NCC2(C)CCC(NC(c3cncs3)=O)C2)cc([N+](=O)[O-])ccc1CO C1(NC(CC2(C)CC2)=O)CC2(CCN(C(c3n[nH]c4c3CCOC4)=O)CC2)C1 C(=O)(CCCC(F)(F)F)NC(C(C)NC(C(n1c(C)ncc1)C)=O)(C)C C(=O)(CCC(C)(C)N(C)C)N1CCC(NC(c2c(COC)nn[nH]2)=O)C1 C1(CC)CCC(C(=O)NC(CNC(=O)Cn2cc(Br)c(C)n2)CCOC)CC1 N1(C(c2c(Br)cc(C)s2)=O)CC(C)(C)CC1CNC(=O)CC(C)O C(=O)(CCCP(C)(C)=O)NCC1(C)CCCC1NC(c1cc(F)cs1)=O C1(C#N)(C(N(C2(CC(=O)N(C)Cc3ncnn3C)CC2)C)=O)CC2CC2C1 C(=O)(C1=NOC(C)C1C)N1CCC(NC(c2c(SC)cccn2)=O)CC1C CC1CN(C(=O)CCc2nncn2C)CC1(C)CNC(=O)C1=COCCO1 N1(C(c2cnc(SC)[nH]2)=O)CC(NC(c2cc(C)n(C)n2)=O)C2CC12 c1(CCNC(C(=O)NN(C2CCCO2)C2CC2)=O)ccc2ncsc2c1 C1(C(N)=O)CN(C(C2CC(C3CC3)=NO2)=O)CCC1NC(C1CC12CCSCC2)=O c1(CC(=O)OC(C(=O)OC)CSC)cc(C=C(C)C)ccc1OC N1(C(CC2CCC(C)(C)CC2)=O)CC2(C1)SCCC2NC(C1C2CC3C(C2)C13)=O C1(CNC(CCS(C)=O)=O)CCC2CN(C(=O)CCCc3cc[nH]n3)CC12 c1(C(=O)NCC(C)(C)NC(C2CCCCC2O)=O)ccc(F)c(F)c1F N1(C(C(C)Sc2ccccc2)=O)CC=C(CNC(=O)C2=CCSC2)CC1 c1(OC)cc(-c2nc(CCOC)nn2-c2ccc(F)nc2F)ccc1Cl c1(-c2nnc(N(C(CCC3C(C)CCC3)=O)C3CCCC3)s2)ccc(S(C)(=O)=O)[nH]1 C1(C(N2CC(NC(c3ccc(Cl)o3)=O)(CO)C2)=O)Cc2ccccc2CO1 C1(CCOC(C)C)CCCCN1C(c1c[nH]nc1O)=O.C(C(=O)NCC)SCCC c1(CCC(=O)NCC2CCC(NC(=O)Cc3ccns3)CC2)cc(F)cc(F)c1 CC1(C)COCC(CS(=O)(=O)NC(c2ccccc2Cl)CO)O1 c1(CCCCC)ccc(C(N2CC(C(C)NC(=O)CC3CCC(C)O3)C2)=O)s1 C#CCC(CC#C)C(=O)N(C1CN(C(c2ccn(COC)n2)=O)CC1(C)C)C C(=O)(C1=C(Cl)CCCC1)NCC1CN(C(COCCC#C)=O)CC12CC2 N1(C(=O)CCCOc2ccccc2)CCn2c(cnc2CC(F)(F)F)C1 C(=O)(C1=NOC(C)C1)NC(CN(C(c1c(C)cc[nH]1)=O)C)C c1(C(=O)NCC2C(NC(c3c(CC)cno3)=O)CC2)c[nH]c2nccc(Br)c12 C1(CCC)CN(C(=O)C(CC)C(C)C)CCN1C(c1ccc(O)c(F)c1)=O C1(NC(C(C)OC2CCOCC2)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 C1(C(N2CC=CC(NC(=O)C(O)C(F)F)C2)=O)C2CCC3(COC(=O)C13)O2 CC12COC(C(=O)NCCCC3(NC(C4(C)C=CCCC4)=O)CC3)(C1)C2 CC1SCCCC1C(=O)N(CCCNC(=O)C(C)(C)C1CCC1)C c1(C(N2CC3C(C(N4CC5C(C(=O)OCC)C5C4)=O)(C3)C2)=O)cc2ncccn2n1 c1(C(N(CCCNC(C(C)CF)=O)C)=O)ccc(-n2cccc2)cc1O c1(CO)cscc1C(F)F.c12ccc(o1)CNC2c1nnnn1Cc1cccs1 C(=O)(CC1=CCOCC1)N(CC(=O)NCC(O)CF)CCC C(=O)(CCCN(C)N=O)N1CCCC(N(C(c2ccc(F)cc2N)=O)CC)CC1 c1(C(N2CCC(N(C(c3nocc3C)=O)CC)CC2)=O)cc(OC)cc(C)c1 N1(C(C(CC)NC(N)=O)=O)CCC(c2cn(C(C)C)nn2)C12CC2 N1(C(C(CCC)OCC)=O)CC2(CCCC(CNC(c3cnsc3C)=O)O2)C1 C1(C(=O)NC(c2cn(C)nc2)c2ccccc2)C2CS(=O)(=O)CC12 C1(CNC(Cc2c(CC)cccc2)=O)CC2CCC(C1)N2C(c1nccn1CC)=O c1(CC)nn(C)cc1CNC(=O)C(C1CCCC1)NC(=O)C=Cc1nccs1 CC1CC(CNC(=O)CC(=O)NC2CC2)CN1C(=O)CCn1cc(Br)cn1 Cc1ccc(CCC(=O)NC(c2ccccc2)CNC(=O)CCc2cccs2)o1 N1(C(C(=O)NC(c2ccc(-n3ccnc3)cc2)C)=O)CCCC(NCCSC)C1 C(=O)(CC(C)(C)C)NCC(=O)NCC1CC(NC(C(c2ccccn2)C)=O)C1 c1(C(N2CCC(OC)(CNC(=O)Cn3cccn3)C2)=O)cc(P(C)(C)=O)cs1 CCCCC(C(=O)NCC1(O)CC(NC(c2ccc(F)cc2O)=O)C1)N(C)C c1(C(N2CC3(OCC(C(=O)NCC4CC(=C)C4)C3)C2)=O)c[nH]c2ccccc12 N1(C(C(C2CN(C(=O)C(C)CO)C2)OCC)=O)CCCC1CCN(C)C c1(C(=O)NC2C(CC)N(C(=O)CCc3cccs3)CC2)cnc2sccc2c1 c1(C(=O)NC(CNC(C(CC=C)C(C)C)=O)C(C)C)c[nH]c2ccccc2c1=N CCC(C)(C)C(C)CC(=O)NC1CC2CCC1N(C(C1COC1)=O)C2 Nc1cccc([N+](=O)[O-])c1C(N1C2CCC1CC(NC(C1(CCF)CC1)=O)C2)=O c1(SC)ccc(CC(=O)NC(C)(C)CNC(=O)CC2CC2)cc1 C1(C(=O)NCCC(C)NC(c2cscc2Cl)=O)CNC(=O)N1C Cn1nc(Cl)c(C(=O)NC2CC(C)(NC(=O)C(c3ccc(Cl)cc3)=O)C2)c1Cl C1(C(C)(C)C)C(=O)N2CCSCC2C(=O)O1.CC(C)CCNCCC(=O)O N1(CC(N2CCSC3(CCCC3)C2)=O)C(=O)NC2(CCC(C(=O)O)CC2)C1=O C(=O)(C#CC1(C)CC1)NC1CC(CNC(c2cccc(N(C)C)n2)=O)OCC1 N1(C(C(C)N2CCC2)=O)CCC(CNC(C2OCC2(C)C)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CC=C(CNC(C(C)(C)c2ccccc2)=O)CC1 CC(C)C(CNC(=O)C(C)CC1CCCCC1)NC(c1cc(CN(C)C)on1)=O c1(C(N(CC(O)CNC(C2(C)CSC2)=O)C)=O)cc2nc(F)ccc2o1 c1(OC)cncc(C(=O)NCC23CC2CN(C(C2CC2c2cnc[nH]2)=O)C3)c1C C1(C(=O)NCCCC2(NC(=O)C=CC3CCC3)CC2)CCCCC12CCC2 C(CCCCC(=O)NCCC(C)(C)NC(c1nc(C)n(-c2nc[nH]n2)n1)=O)SC C1(N(C(C2CC(O)(CC#C)C2)=O)C)CCC(NC(c2cn(C)c(C)n2)=O)CC1 N#Cc1cccc([N+](=O)[O-])c1NC(CNC(c1cccc2oc(O)nc12)=O)C1CC1 C1(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)CN(C(C2CC(C)(F)C2)=O)CC1C O=C(CC1OCc2ccccc21)NC1CCC(NC(c2sccc2Cl)=O)C1 C(CC(CC)C(=O)NC1CC1CNC(c1cncc(-n2cnnn2)c1)=O)=CC C(=O)(C1Cc2c(Cl)cccc21)N(C1CCN(C(c2c(C)occ2)=O)C1)C c1(C(=O)NC(C)CC(C)NC(=O)CCCc2cnn[nH]2)cncc2c1CCCC2 c1(C(N2CC(CNC(C3(CC(C)=O)CCC3)=O)OCC2)=O)ccc2nc[nH]c2n1 n1(CC)cc(Cl)c(C(=O)NCC2CC(NC(c3nnn(C(C)C)c3C)=O)C2)n1 C(C)(C(=O)N(C(CO)C1CC1)C)N(C(C)=O)C.C12(CC1)C(=O)O2 c1(C(N2CCC(CNC(C3=C(C)CCC3)=O)C2)=O)ccc(F)c(F)c1O Cc1nc2cc(C(=O)NC(C)CCNC(=O)CNC=O)ccc2o1 c1(C(CC)C(=O)N2CCCC2Cn2nnnc2-c2ccccc2Cl)ccc(F)cc1 c1(COC)cccnc1C(=O)NC(CNC(c1csc(CC(C)C)n1)=O)CO Cc1csc(C(C)C(=O)NCCCC(C)NC(=O)CC2(CC3CC3)CC2)n1 c1(C(=O)NCC(C)NC(=O)C=Cc2cccc(Br)c2)ccc(N)cc1F c1(C(=O)NCc2ccc(C(N)=O)s2)cc(-c2ccco2)n(-c2ccccn2)n1 Cn1cc(CNC(C2CC(CNC(=O)C(F)CC3CCCC3)C2)=O)c(O)n1 N1(C(Cc2c(Cl)cn(C)n2)=O)CCC2CC2(C(N2CC3C(C(N)=O)C3C2)=O)CC1 C1(CNC(CCOC(C)=O)=O)CC(O)C(O)CC1C(=O)N(CCCO)C1CC1 c1(C(N(C(CN(CCCC#C)C)=O)CCCCCCC)=O)nccc2[nH]ccc12 CC1CCC=C1C(=O)NC1C2CC1CN(C(=O)COc1ccccc1Cl)C2 Cc1cc(C)cc(C=CC(=O)NCC(O)CCNC(c2ccnc(C)c2)=O)c1 Cc1c(C(N2CC(C(=O)Nc3cn(C)nc3O)C(F)(F)C2)=O)cccc1F C(=O)(C(F)CC(C)(C)NC(=O)Cn1nc(C)nc1C)NC(C(CCC)C)C C(=O)(C(C)(C)CC(C)(C)C)NCc1c(CN(C)C(c2nocc2Cl)=O)cccc1 Cc1cccc(-c2cnccc2C(N2CCCC2c2cccnc2)=O)n1 O=C(C1=COCCC1)NC12CC(C1)N(C(=O)Cc1ccc(F)c(Br)c1)C2 c1(CCN(C)C(C2OCCC2NC(=O)Cc2cnsc2)=O)ccncc1 C1(C(=O)NC(CC)CNC(=O)C(C)N(CC)CC)CC(C)(C)OC1(C)C c1(C(c2nccs2)NC(N(C)CCOC(F)F)=O)ncncc1N c1(NC(C2N(C(C3CC(=C)C3)=O)CC3(CC3)C2)=O)nc(Cl)c2c[nH]nc2n1 C(CCCC(CO)N)NC(C(CN(C)C)(C)C)=O.C(=O)(C#CC(C)(C)C)N c1(C(C)=O)cccc(C(N2CCOC(C(C)NC(=O)CNS(=O)(=O)NC)C2)=O)c1 C(c1cncn1C)=CC(=O)N(C(C)C(N1CCC(CC2CC2)C1)=O)C N1(C(Cc2cc(C)ns2)=O)CCC(C(C)(C)C)(CNC(C2COC(=O)N2)=O)C1 c1(CC(C(=O)NC)NC(c2csc(C(C)C)n2)N2CCCCC2)ccc(F)cc1 c1(C(N(C)CC2CCN(C(CC(CC)OC)=O)C2)=O)cc2c(nc1N)CCCC2 C#CCC(C)C(=O)N1CCCC1CNC(c1ncoc1-c1ccccc1)=O c1(NCC(C)C)ccc(S(=O)(=O)NC2CC2C2CC2C)cc1C#N n1(CCCNC(C2CC(C)C(C)CC2)=O)cnc2ccc(F)cc2c1=O N1(C(C(c2onc(C)n2)(F)F)=O)CCC(CCn2cc(C(=O)O)cn2)CC1 C(C(F)C(=O)N1CC(C#N)C1)C1CN(C(C2CN(C(C)=O)C2)=O)C1 c1(C(=O)NCC2N(C(c3[nH]cc(C)c3C)=O)CCCC2)ccc(F)c(I)c1 C(=O)(C1Cc2ccccc21)N1CCC2CC(C(N(C(C)C)CCC(F)(F)F)=O)C2C1 N(C(=NCCc1ccccc1O)NCC1CC1)C1CCCC(CC#N)C1 C1(NC(C2CN(C(C3(CO)CCOC3)=O)CCO2)=O)CCCC2(CCC2)C1 C12(NC(c3nn(CC)c(C)c3)=O)CCCC1N(C(=O)CCOCCCOC)CC2 N1(C(c2cnn(CCC)c2C)=O)CCCC(N(C(=O)CS(=O)(=O)NC)CC)CC1 CCC(O)C(C)C(=O)NC1CC2CC(NC(C3(CO)COC3)=O)C2C1 C1(F)(C(N(C)CC2CCN(C(c3cc(CC)n(C)n3)=O)CC2)=O)CCS(=O)(=O)C1 C1(CNC(=O)CCOc2ccccc2F)CN(C(C23COCC2C3)=O)CCCO1 C1(C(=O)NC(c2cccc(F)c2)C2C(C(C)(F)F)C2)CN(S(N)(=O)=O)C1 c1(C(=O)NC23CC(CC(=O)NC(C)C(F)F)(C2)C3)ccc2ncccc2c1 N1(C(CCC(=O)NCC)=O)CCN(C(c2c(C)ccnc2C)=O)CC1C1CCC1 c1(C(C2(C)CCS(=O)(=O)C2)C)cc(Br)ccc1S(=O)(=O)NC1CC1(F)F c1(OC)cc(=NC(=O)C2C3CCN(C(C4(C)CC=CC4)=O)CC23)[nH]n1C C1(C(N2CC3(CCCC3)C2)=O)(NC(CSCC)=O)CCC(C)(C)C1 Cc1cc(Br)c2[nH]c(C(=O)N(C(C)CNC(=O)CC3(C)CC3)C)cc2c1 C#Cc1c[nH]nc1C(=O)NC1COCCC1C(N1CCC12CCCC2)=O CCCCCCCCCS(=O)(=O)N1CC2OCCC2CN1C C(C(C)(C)CNC(C1CCCC1NC(=O)CN1CCCC1)=O)OC C1(CCC)C(C)CCCN1C(=O)C(CNC(c1ccsc1)=O)N(C)C N#Cc1ccc(C(=O)N(CCNC(C2CC2c2ccccc2)=O)CC2CC2)c(F)c1 C1(C)(C(=O)NCCOC2CCN(C(C(C#C)(C)C)=O)C2)CCCCNC1=O c1(-n2cc(-c3nc(CSC)nn3-c3ccc(F)c(Cl)c3)nn2)ccc(S(C)=O)cc1 C1(NC(CN(C(C)=O)C)=O)CCN(C(C2CC3CCC(C2)O3)=O)CC1O Cc1cc(C(=O)NC2(CO)CC(F)(F)C2)c(F)c(Br)c1 C1(NC(C=C(CC)CC)=O)CN(C(=O)C(C)=CC2CC2)CC1c1ccccc1 c1(-n2c(-c3[nH]c(=NC)sc3)nc(COC)n2)ccc(Cl)c(OC)c1 N1(C(CCCCCCCC)=O)CCC2(CCN(C(=O)COCCF)CC2)C(C)C1 n1(CC(=O)NCC(CCCC)NC(C2(Br)CC2)=O)nc(C)c(Cl)c1C c1(OCC)ccc2cc(C(c3nnnn3C)N)oc2c1.C1(C)(CF)CCC1 C1(C)(CNC(C2(C)CCSCC2)=O)COCCN(C(C2CC(F)(F)C2)=O)C1 Cc1nc(N2CC3CC2C3C(=O)NCC2CCC2)c2c[nH]nc2n1 N1(C(C2N(C(=O)OCC)CSC2)=O)CCOCC1CCNC(=O)C(F)F [N-]=[N+]=NC1CCC(C(=O)NCC(O)CNC(=O)CCNC(C2CCC2)=O)CC1 Cc1ccc(N2CCCC2)cc1.N(C(=NCc1ccccc1)NCC(F)F)C1CNC1 C1(CC=C)(NC(c2csnc2C)=O)CCN(C(C2CC3C=CC2O3)=O)CC1 Cc1cc(C)c(C(N2CCCC(CNC(=O)CN(C)C)C2)=O)c(=O)o1.C(=O)C(C)C Cc1cc(C(=O)NCC2CN(C(=O)CN(C3CCC3)C)CCN2C)ccc1O CC1CN(C(C2CCCOC2)=O)CC(C(=O)Nc2ccc(Cl)cc2)O1 C1(C2CCCCC2)(NC(C2N(C(c3c(CC)nns3)=O)CC(O)CC2)=O)CC1 Cc1ccc(F)c(C(=O)NCCCC2CCCN2C(=O)C(C)OCCC(C)C)c1 N1(C(c2cnc3nc(C)oc3c2)=O)CCC2CC(NC(=O)CC(C)C)CCC2C1 C=CC1CCN(C(C2CCCC2CNC(c2ncn(CC)n2)=O)=O)CC1 c1(NC)c(C(=O)NC2CC(F)(CNC(=O)CN3C(=O)CCC3=O)C2)cccc1F C(=O)(CC(O)(CC)c1ccccc1)NCCCNC(COCC)=O c1(C(N2C(CNC(c3c(SC)cccc3)=O)C(C)CC2)=O)cn(C)c(=O)cn1 CC(C)(C(=O)N1CCC(N(CCO)C(c2cc3sccc3[nH]2)=O)C1)S(C)(=O)=O CCC(CC)=CC(=O)NC(CNC(C1CC1(F)F)=O)CO C(=O)(C1=CCCCC1)NC12CC(NC(C3N(C(=O)OC)CCC3)=O)(C1)C2.C1CO1 C1(C(=O)NC(c2ccncn2)C)CC2(CCC2)CN1C(=O)CC1=CCCCC1 C(CCC(c1ccccc1)NC(c1sccc1OC)=O)NC(C1C(=C)C1)=O N1(C(C=NOC)=O)CCCC(CCNC(C2CCC(N(C)C)CC2)=O)C1 CCCCC(CC)CC(=O)NC(C)(CNC(=O)C(F)C1CCOC1)C1CC1 C(=O)(CCCC(C)(C)C)N1CCC(C)(NC(CC2(C(=O)OCC)CCC2)=O)CC1 CN1CC(F)CC1C(N1CC(O)(CCNC(c2cccc[n+]2[O-])=O)C1)=O N1(C(c2c(C)occ2)=O)CCC(C(F)CNC(c2ccoc2C2CC2)=O)CC1 c1(C(=O)OC)cc(N2CC(O)(C(C)NC(=O)C(CC)SC)C2)n2nc(C)cc2n1 CC1CCCCN1CC(N1CC(F)CC1CC(=O)NC1(C(F)F)CC1)=O C1(OC)CCCN(C(=O)C(Cn2ccnn2)NC(=O)C(F)=CC2CC2)C1 N1(c2nc(C#N)c(Cl)s2)CCCC2(NC(=O)Cc3nc(C4CC4)cs3)CCCC12 n1(CC(=O)N(CCN(C(C2(CC#C)CCCCC2)=O)C)C)ccc(=O)c(O)c1C O=C1CC(C(N2CC(NC(=O)CSc3ccncc3)C2)=O)CCN1 N1(C(CC2C=NN(C)C2=O)=O)CCC2(CC1)CN(C(=O)CCc1cnn(C)c1)C2 C(CN=C(NCC1C(C)(C)C1(C)C)NC(c1cnnn1C)C)OCC=C C1(C(=O)NC(CC)CO)CC(CC)CCN1C(=O)COCCCF C=CC1(C(N2CCC(C(=O)OCC)C2)=O)CCN(C(=O)C(C)N2CCCC2)C1 c1(CNC(C2(CCCC)CCC2)=O)ccc(CNC(C2C3COCC23)=O)cc1F C(=O)(C(C#N)C(C)(C)C)N1CC(CNC(C(CC)N(CC)CC)=O)OCC1 CC1(C)CN(C(=O)C2=CCN(C(=O)Cc3cccnc3)C2)CC(=O)N1 N1(C(Cc2ccc(C)s2)=O)CCN(CCNC(C2C(C)(C)C2(F)F)=O)CC1 C1(NC(c2c(CC=C)cccc2)=O)CCCCCN(C(=O)C=C(C)C(C)(C)C)C1 c1(C(=O)OC)ccc(NC(c2scnc2-c2cc(Cl)ccc2OC)=O)cc1Br c1(N(C2CCNCC23CC3)C(C2CN(CCO)CCO2)=O)ncnc2c1CCC2.C C=Cn1nccc1C(=O)NC1CCC(NC(=O)C(C)n2cncn2)C1 C1(NC(C2N(C(C)C)CCC2)=O)CC2CC(C1)N(C(c1cnn3ccsc13)=O)C2 N1(C(c2c(O)nc(CC)c(C)c2)=O)CCC2CCN(C(c3csnn3)=O)C2C1 C#Cc1cccc(C(N2CC3CC(C2)C3NC(c2cccc(C)c2O)=O)=O)c1F C(C)(CC(F)(F)F)N(C(c1nc(C)[nH]n1)CC1CCCCC1)C(=O)OC(C)C c1(C(=O)NC(C2CCCN(C(=O)C(C)C)C2)C)ncncc1N(C)C Cc1ccc(Br)c(C(=O)NC(CNC(c2cc[nH]c(=N)c2)=O)CO)c1F O=C(C1=NOC2(CCN(C(c3ccccc3S)=O)C2)C1)Nc1cncnc1I Fc1cccc2c(=NC(Cc3cccs3)Cc3ccco3)[nH]c(Cl)nc12 c1(C(N(CC(C)CNC(C2(CO)CC2(F)F)=O)C)=O)c[nH]ccc1=N C1(C(=O)NCC2(CO)CC2)(OC)CN(C(=O)C(C2CCC(=O)N2)C)C1 N1(C(c2c(C)sc(Br)c2)=O)CCN(C(C2CCCC2C)=O)C2CCCC12 c1(CC(=O)NC2CN(C(C)=O)C(C)C2)ccc2c(c1)OCO2.C12CCOC1CC2=O C12CC(CC1O)N2.N1(C(=O)OC(C)(C)C)CCC(c2cc[nH]n2)CC1.C(C=O)O C1(NC(CN2CCC(C)CC2)=O)CC2(CCN(C(=O)CC3CCS(=O)(=O)C3)C2)C1 C1(C(=O)NCC2(CNC(CN(C)CC)=O)CC2(F)F)CC(C)CC(=O)N1 c1(C(N(C2CCN(C(C(CC)C)=O)C2)C)=O)nc2ccccc2s1 c1(OC)cccc2c1OCC(C(=O)NC(CSCC(F)(F)F)C(=O)O)C2 c1(C(=O)NCC2C(NC(c3[nH]c4cc(C)sc4c3)=O)C2)sc2ccccc2c1Cl c1(C(=O)NCCC(C)(C)NC(=O)CCF)c(Br)nc2n1CCCC2 c1(C(=O)NC2C(NC(C(CC)F)=O)CCCC2)c[nH]c2nccc-2c1C C12CCC(C1)NC(=O)C2.c1(C(N(C)CCC2CC2)=O)ocnc1C1CC1 c1(C(C)(C)C)conc1C(=O)NC1CCC(NC(=O)Cc2cccs2)C1 C1(C(N2CCC(CCC(=O)NC(c3ncc[nH]3)C)C2)=O)CCC(O)CC1 O(N(C(=O)C1CCCCN(C(=O)CCC(C)CC)C1)C(C)C)CC c1(OC)nn(C)c(Br)c1C(=O)N(C)CCNC(c1c[nH]nc1C)=O CCCCCCC(=O)NCC1CC1NC(C1(c2ccccc2F)CCC1)=O C(=O)(C(C)(C)C(C)(C)O)N(C(CC(=O)NCCC1CCCC(C)C1)(C)C)C C12(C(=O)NC(CC)CN(C(=O)Cn3cnnn3)CC)CC(C#N)(C1)C2 C(=O)(C1=NN(CCO)C(=O)CC1)N1CCN(C(CC2CC(C)C2)=O)CC1CCO N1(C(CCOC)=O)CC(O)CC1CNC(c1cnc(-c2ccccc2)nc1)=O c1(NC(C2(C)CCN(Cc3cccc(I)c3)C2)=O)c(Cl)cccc1I C1(NC(c2csnn2)=O)CC2CCC1N2C(c1cncc(Cl)c1Cl)=O c1(CC)nc(C)c(C(N2CCC(C)C2CNC(=O)CCC(F)F)=O)s1 N1(C(C2(C)CC(C)C2)=O)CCCC(C(=O)N(C2(CO)CC2)C)C1 CCCC(C)(O)CC(=O)NC(CO)C(C)NC(C1CCCC1C1CC1)=O C1(CCC(=O)NCCC(C)N(C(CCCOC(C)C)=O)C)CCCCN1C C1(C(N(C(C)C(=O)N(C)Cc2cccs2)C2CC2)=O)CC2(CC2)CO1 c1(C(N2CCC(COC)C2)C(=O)NC2(C)CC2)csc2c(Cl)cccc12 c1(C(N2CCCC(NC(C(CN(C)C)(C)C)=O)C2)=O)noc2ncccc12 c1(C(N2CC(C)(NC(CCOC)=O)C2)=O)ccc(OC2CCOC2)cc1 C(=O)(C1CCc2nccn21)NCC(C)(C)NC(C=C(COC)C)=O c1(C(c2nnnn2C(C)C)NC(CC)C2CC2)c(F)cc(F)c(Br)c1F C(=O)(C(O)CCCNC(C1(C#N)CCOCC1)=O)NC1C(C)CN(C)C1 c1(CN(C(C2CCOCC2)CC)C=O)ccc(C)c(Br)c1 CCC(CC)CC(=O)N1CCCC(O)(CN(C)C(C2CC(=C3CCC3)C2)=O)C1 CC(C)(C#N)CCC(=O)NC1CC1NC(c1ccc(-c2ccncc2)c(F)c1)=O c1(C(N2CCC(O)(CCNC(C=C(CC)C)=O)C2)=O)cc(C)cc(O)n1 c1(C(NNC(=O)C2N(C)CCC2)=O)ccc(N)cc1 C1(CNC(C2CC(CC3CC3)C2)=O)CN(C(C2(CCO)CC2)=O)CCC1(F)F C1(NC(c2c(OCC)cccc2F)=O)COC2CN(C(=O)CNS(N)(=O)=O)CC12 c1(NC(CC2C(CNC(C(=O)NCC)=O)C2)=O)cn(C)c(=O)nc1O C12(NC(C3(NC(C)=O)CCC3)=O)CCCC(CN(C(c3ccc[nH]3)=O)C1)C2 c1(C(N(CC(C)O)CCNC(COC)=O)=O)c(C)c2ccc(F)cc2oc1=O C(=O)(CC(C)(O)C=C)CC#C.C1(N)CCN(C(C2(COC)CC2)=O)CC1 N1(C(C(c2cccnc2)OC)=O)CCC(C)C(CNC(c2cc(C#N)on2)=O)C1 N1(CCC(=O)NCC(C)(CO)NC(Cn2cc(C)nc2)=O)CCCCC1=O C1(C(N2CCC(NC(C(CC(C)C)F)=O)CC2)=O)Cc2cccnc2C1 c1(C(=O)NC(CC)C(OC)OC)nc(C)n(-c2ccc(Cl)cc2)n1 N1(C(=O)OC)CCCC(CNC(C2CN(C)CCO2)(C)OC)C1 c1(C(N2CCOC(C3CCCOC3)C2)=O)ccc(Br)c(Cl)c1F Cc1cc(F)ccc1C(O)C(=O)NC1CCC(NC(=O)C(C)n2cncn2)CC1 c1(C(=O)NC(CNC(=O)CCc2cscn2)C2CC2)cc2sccc2s1 c1(CNC(C2CCCN(C)C2)=O)cccc(Br)c1OC(F)F.N1(C)CC1 C1(CNC(Cc2c(C)n[nH]c2C)=O)COCCN(C(C2CCCCC2)=O)C1 C#CCC(C(=O)N1CCC1(C)C(C)C)NC(=O)Cc1cc(C)n(C)n1 N1(C(c2c(C)ccnn2)=O)CCC(NC(=O)C(N2CCOCC2)C)C(CO)C1 N1(C(c2cc(OC)nn2C)=O)CC2CC(NC(C3C(CO)C4CCCC34)=O)C1C2 CCC(C(=O)NCC1CC(F)(CNC(c2cccc(F)c2)=O)C1)C(C)O C(CN=C(NCC(Cc1ccc(Br)cc1)CO)NCC1CC1)NC(C)=O N1(CC(=O)NCC(C)CN(C)C(c2c[nH]nc2C2CCC2)=O)CCSCC1 C1(N(C(C2CN(C(=O)Cn3ccc(C4CC4)n3)C2)=O)C2CC2)C2CC3C(C2)C13 N1(C(c2c(C)onc2)=O)CC2CN(C(C3CCCCN3C)=O)CC2(C)C1 C(C(=O)N1CC2CCC2C1)(C(C)C)NC(C1C(COC)OCC1)=O N1(C(C2CC(O)(CC#C)C2)=O)C2CCC1CC(NC(=O)C(C)C(C)O)C2 c1(SCC(=O)NC23CC(NC(C(C)NC(CC)=O)=O)(C2)C3)nc2ccccc2o1 c1(C(=O)NC2CN(C(C(CC)=O)=O)CC(C)C2)cccc2cccc(C)c12 c1(C(=O)NCC2CCN2C(=O)C(F)n2ccnc2)cncc2sccc12 Clc1cc(Br)ccc1C(c1nnnn1C1CCCC1)Nc1cncnc1OC CCC(CC(=O)NCc1cc[nH]c1C(=O)NC1CC2C(C1)C2(F)F)C(F)F C#CC1CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CCN1C(C1CC2CCC1CC2)=O C1(C2CN(C(C3(CO)CCCO3)=O)C2)(NC(c2c(CC)n(CC)nc2)=O)CC1 c1(CC)cn2c(n1)CC(C(=O)NCC(CC)NC(c1ccnc(O)c1)=O)CC2 N1(C(C(COCC)N(C)C)=O)CCCC(C(=O)NCCc2cncs2)C1 c1(C(C)(C)C)ccc(Br)cc1OC(=O)CCc1cccc(Br)c1 c1(NCc2cccc(C)n2)nccc(=NC2CC3(CCOC3)C2)[nH]1 N1(C(C(=O)NCC)=O)CCN(C(=O)C(O)CC2CCOCC2)CC2CCCCC12 CC(C)CC(C)C(=O)NC(C)CCN(C)C(c1cc(O)ccc1Cl)=O C1(N(C(CSCC)=O)C(c2nnc(C3CC3)s2)=O)CCCC1C(=O)OC C1(CNC(c2c(CC)cccc2)=O)N(C(C2COC(=O)N2)=O)CCCC1(C)C C1(C(=O)NCCCCCNC(c2n(CC)nc(C(C)C)c2)=O)C2CS(=O)(=O)CC12 CC(CCC(C)(C)C)C(=O)NCCCCN(C(=O)C=Cc1cccn1C)C CN1CCC(F)(C(=O)NCCCCN(CCCNC(=O)CCn2ccnn2)C)CC1 N1(C(c2cc(COC)no2)=O)CC(CNC(C2(C(F)(F)F)CCC2)=O)C(O)C1 C1(CC(=O)N(CC(C)C#N)C)CC2(C1)CN(C(C1(C(F)(F)F)CC1)=O)C2 N1(C(C(COC)O)=O)CCCC1(C(=O)NCC(N1CCOCC1)=O)C(C)C C1(CNC(CC(C)CF)=O)CCC(C)(C)CN1C(c1ccsc1)=O N1(C(CNC(CCC)=O)=O)CCCC(CNC(=O)Cc2cccc(C)c2F)CC1 c1(OC)ccc2nc(NC(=O)CSCc3c(I)cnn3C)[nH]c2c1 c1(C(=O)NCC2CN(C(c3cnc(CCCC)s3)=O)C3C2C3)cnc2n1CCS2 C12CC13CC(C3)NCC(=O)N2.c1(C(C)C(=O)OC(F)F)ccccc1.[SH](=O)(=O)C C1(CC)CCN(C(=O)CC2CCCCC2N(C(c2nccnc2C)=O)CC)CC1 C(C1CC1)(C1CC1)=CC(=O)NCC1CCN(C(COC2(C)CCCC2)=O)C1 c1(C(N(C)CC2(O)CN(C(C3C(SC)CCC3)=O)C2)=O)c(F)ccc(F)c1O c1(CC)nc2ccc(NC(c3nnnn3C(C)C)C3CCCOC3)cc2s1 c1(C(N2CCC(NC(C3(C)CC=CC3)=O)C(CO)C2)=O)ccc2cnnn2c1 C1(C(=O)NCC(C)(C)CNC(=O)Cn2nnc(=O)[nH]2)(OC)CCOC1 c1(CCC(=O)NC2CCN(C(c3csnn3)=O)CC2F)ccc2c(c1)OCCO2 CC1OC(=O)NC1C(N1CCC(C(N2CCCC23CC3)=O)C1C)=O c1(C(N(C2CCN(C(C(C3CC3)SC)=O)C2)C)=O)nc(C)[nH]c1C(F)(F)F c1(CNC(C(COC)COC)=O)cc2n(n1)CCN(C(C1CCCC1(C)C)=O)C2 C(=O)(CCC(C)CN(C)C)NCCCOC1CCN(C(C(CC)(C)O)=O)CC1 C(=O)(CC1OCc2ccccc21)NCCCCCCNC(CC(C(CC)(C)C)C)=O c1(CC)ccc(C(N2CCN(C(c3ccc(F)c(C)c3)=O)CC2C)=O)cc1Br c1(C(N2CC(C)(NC(CC3C(C)CCC3)=O)C2)=O)cnc2c(c1)CCOC2 Cc1cc(C(N2CCC(CNC(=O)CCC(C)N(C)C)C2)=O)ccc1Cl C1(CC(=O)N(CC)CC2CCNC2=O)CCN(C(C)CCO)CC1 CN1CCc2cc(C(=O)NC3CCOCC3NC(c3ccco3)=O)ccc21 c1(COC(c2cccc(-c3n(CC)nnn3)c2)=O)ncc(F)cc1F CC(C)(C)C#CC(=O)NCCC(O)C(=O)N1CCC(CC(N)=O)CC1 C=CC(C)(CC)C(=O)N1CCCC(NC(c2ncn(C(C)(C)C)n2)=O)C1 C1(NC(C(COC)(C)OC)=O)CN(C(=O)C2=NOCC2)CCC1C(F)(F)F N1(C(C2C3(CCN(C(CN(C(=O)OC)C)=O)C3)C2)=O)CCC2(CCCOC2)C1 S(=O)(=O)(c1ccc(Br)cc1NCCCCCCOC)N1CC(CC)NC(=O)C1 O=C(C)CCCCN=c1cccc(S(=O)(=O)NCC2OCC3CCC2C3)[nH]1 C1(C(=O)NCC(=O)OCC=C)CCN(C(C2CCSC2)=O)C(C)(C)C1 N1(C(CCC2C(C)(C)C2)=O)CC(C=O)C(F)(F)C1.C(C(C)(C)O)(C1CC1)NC(C)=O C(=O)(C(C)(COCC)CC)NCC=C(C(N1CCCC(CC=C)C1)=O)C C1(NC(c2c(C)ccc(OC)c2)=O)CN(C(=O)CC2(CSC)CC2)C2CCCC12 N1(C(C(C)(Cl)Cl)=O)CC(C(=O)NOCC(F)(F)CC2CC2)C(C)(C)C1 C1(COC)CC(CNC(c2n[nH]cc2C(C)(C)C)=O)N(C(=O)C(C)SC2CC2)C1 N1(C(c2cnsc2)=O)C2CCC1CN(C(c1cc(C)c(OC(F)F)cc1)=O)CC2 N1(C(CCc2n(C)nnc2)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C2COCC12 C1(C(=O)NCC=CCNC(=O)C(O)Cc2cnc[nH]2)CC2CCC1C2 c1(C(=O)OC2CCN(C(=O)CCC3CCN(C(C=CC)=O)C3)C2)ccc(O)cc1 C1(C(N2C(C(N3CCC(O)(CO)C3)=O)CC2)=O)CC2CC1CC2O CC1OCCC1C(=O)NCCCN(CCCCNC(c1sccc1CO)=O)C CC1(C(=O)Nc2cc(-c3ccccc3)no2)CCCN1C(c1cccs1)=O c1(C(=O)NC23CCCN(C(CCC#C)=O)CC2C3)nc(C)n2ccccc12 c1(OC)ccc(C(N2C3CCC2CC(CNC(=O)CC2CC2C)C3)=O)c(F)c1N N1(C(c2[nH]cc(C)c(=O)c2)=O)C2CCC1C(CO)N(C(C1(C(N)=O)CC1)=O)C2 N1(C(c2c(C)n[nH]c2)=O)CC(NC(c2c(C)nsc2Br)=O)C(C)(C)C1 C(CNC(C12CC(CC(F)F)(C1)C2)=O)(CCNC(C1(N(C)C)CCCC1)=O)OC c1(COC(C2(CC)CN(C(=O)Nc3ccccc3CC)C2)=O)ccc(F)c(C)c1 C1(CNC(C2(NC(CSCCC(C)C)=O)CCSC2)=O)CCCOCC1 C(=O)(C(O)CCCNC(=O)C1=NNC(=O)C1)NCCCCS(C)=O c1(C(N2CCN(C(c3c(OC)cncc3)=O)CC2C)=O)cc(C)c(O)cc1C c1(C(=O)OC)ccc2c(c1)CCC(NC1CCC(CCl)C1)C2 C1(C(N2CC(C(=O)NCCNC(C3N(C)CC(F)C3)=O)C2)=O)CCOCC1(C)C c1(OCC(=O)NC2C(NC(c3c(C)c[nH]n3)=O)CC2)cccc(S(C)(=O)=O)c1 C1(C(=O)OC)CCC(C)N(C(c2cc(C)oc2C)C(=O)NCCCF)C1 CCC(CC(=O)NCCC(C)N(C)C(C1COC2COCC2O1)=O)C(C)C Cc1ccc(C=CC(=O)NCC2CCCN2C(=O)CC2CC(C(F)F)C2)o1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC=CC1C(=O)N(C1CCCC1(F)F)C c1(CC(=O)NC(C2CCCCC2)C(C)NC(CCSC)=O)ncccc1C Cc1cnc(C(N2CCCC(CNCc3ccc(O)nc3C)C2)=O)cc1Cl Cc1cccc2cc(C(=O)NC(CNc3ncc(Br)c(O)n3)C(C)(C)C)nn12 C1(NC(=O)C(=O)NCCO)CC2CN(C(=O)COCCSC3CC3)CC12 N1(C(C=COCC)=O)CCCC2CN(C(c3c(C)nc(C)n3O)=O)CCC12 c1(C(N(CC)CC2CCCN(c3nc(C)cc(C)n3)C2)=O)cnc2ccccc2c1 Cn1cc(S(N)(=O)=O)cc1C(c1nnnn1CC1CC1)Nc1cn(C)nc1OC N1(C(C2CC3CN(C(C4(N(C)C)CCC4)=O)CC2C3)=O)CCC2(CC1)CC(O)C2 c1(OC)oc(C)nc1C(=O)NC(C)(CNC(c1cc(CN(C)C)c[nH]1)=O)C(C)C N1(C(C(CC)(F)C(=O)OC)=O)CCC2CCC(C1)N2C(=O)Cn1cc(C)cn1 N1(C(c2c(C)[nH]nc2CO)=O)CC2(CCC(NC(C3CC3(C)C)=O)CC2)C1 c1(C(=O)NC(C#CC)C)cc2c(cc1OC)CCCC2 CCC(CC)C(C)C(=O)N1CCN(C(=O)C(C)C)C(CO)C1 c1(SC)ncc(C(N2CCC(CNC(C3COCCN3C)=O)C(C)C2)=O)c(O)n1 c1(OC)cc2c(cc1Br)CCN(CCOc1cccc(OC)c1)C2 c1(CC)sc(=N)[nH]c1C(=O)NCCN(C(c1coc(Br)c1)=O)C1CC1 c1(C(C)=O)cc(NCCC2CC(NC(C3(C)CC3(F)Cl)=O)C2)ccc1[N+](=O)[O-] N1(Cc2ccc(-c3c(N(C)C)cccc3)cn2)CCc2ncncc2C1 C(CCCCCNC(=O)CCCCO)N(C)C(C1CCCN(C(=O)C(N)=O)C1)=O CCC(C(=O)NCCCCC(CO)NC(c1cncc(C)c1)=O)C(F)(F)F N1(C(c2c(N)nccc2)=O)CCC2(CCCC2NC(c2ncc(F)cn2)=O)C1 C(=O)(C#CC1CCN1C(=O)OC(C)(C)C)OC(C1CN(C2CN(C)CCO2)C1)C c1(C(N(C(C)CCNC(c2cccc(C(F)F)n2)=O)C)=O)nc(Cl)ccc1N c1(C(=O)NC2C(NC(C3(CC=C)CC3)=O)CC2)cc(Cl)c(Cl)c([N+](=O)[O-])c1 C(=O)(C1=C(C)CCOC1)N1CC(CC=C)(NC(C2C(C)(C)C2(C)C)=O)C1 C1(CNC(C(CNC(c2cn(CC=C)nc2)=O)C(C)C)=O)CC2(C1)CC21CCC1 C1(C(=O)NCC2NC(=O)OC2)COCCN1C(=O)CCCn1ccnc1 CN1CCC(C(N2C3CC2CN(C(=O)C(CO)N(C)C)C3)=O)CC1=O c1(CC(=O)CN(CCNC(C(C2CCCOC2)OCC)=O)CC)ccccc1Cl C(=O)(CC(F)(F)C(F)(F)F)N1C2CC(CNC(C3NC(=O)C4CC34)=O)CC1CC2 N1(C(C2(C)CC(C)C2)=O)CCC(C)(C)C(NC(=O)CN2CCNC(=O)C2)C1 C(=O)(CCCC(C)(C)C#N)NC1CC(CNC(CC(CC)OC)=O)C1 N1(C(c2n(CC)ncc2)=O)CCN(C(c2coc(O)n2)=O)C(CC(F)(F)F)C1 Cc1cccc2cc(C(N3CCC(NC(C4CC45CCOC5)=O)CC3C)=O)[nH]c12 c1(C(N2C3CN(C(C(F)OC)=O)CC2CC3)=O)cn(C)c2ccc(F)cc12 CCC(CC(F)F)C(=O)NC1CC12CCN(C(=O)CCc1ccccc1)CC2 C(O)(C(=O)N1CC=CCO1)C1CCN(C(CC2(C#N)CC2)=O)C1 C(=O)(CCC(C)(C)C(=O)N1CCC(NC(c2coc(C(C)C)n2)=O)C1)OC c1(C(=O)NCC2OCCN(C(C3N(CCC)C(=O)CC3)=O)C2)n[nH]cc1[N+](=O)[O-] Cc1ccc(C=CC(=O)N(CCCO)C(C)(C)C)cc1C N1(C(=O)NC(c2ccccc2NC(N)=O)C)CC2CC1C2NCc1nc[nH]n1 Cn1ncc2cc(CC(N3CCN(C(c4csc(=N)[nH]4)=O)CC(O)C3)=O)ccc12 CCCC(C(=O)NCC(CNC(c1cc(C(C)(C)C)c[nH]1)=O)CO)OC CN1CCCC1CNC(=O)C(c1ccco1)NC(=O)C(O)c1ccco1 Cc1cc(S(C)(=O)=O)ccc1NC(c1cccc(C(F)F)c1F)=O c1(C(=O)NCC(CNC(CC(CC)C2CC2)=O)F)cnc2cc[nH]c2c1 Cc1cc(C(=O)NCC2CCCN2C(=O)C=CC=C(Cl)Cl)c2sc(=N)[nH]c2n1 CC1(NC(c2nccnc2Cl)=O)CCCN(C(=O)C(O)CC2CCCCC2)C1 C(=O)(C(C)C(C)NC(=O)CC1(OCC(=C)C)CCC1)NCCOCC C(=O)(CC(C)P(C)(C)=O)NCC1(NC(c2c(C)nc(CO)o2)=O)CCC1 C1(C(C)=O)CCCCN1S(=O)(=O)C(F)F.C12CCN1C2=O Cc1nsc(C(=O)NCC2CCC(NC(C3(CO)CCOCC3)=O)C2)c1N CCC(C)CC(C(=O)NCCC(C)CCO)NC(C1CCN1C)=O C1(NC(COCCOCC#C)=O)(CNC(c2noc(C)c2C)=O)CCCCCC1 Cn1cc2cc(CC(=O)NCC3(NC(=O)C4=COCCO4)CCOC3)ccc2n1 CCCCC(C(=O)NCCC1(CO)CCC1)NC(C1CC2CC2C1)=O CCS(C)(=O)=NC(=O)CC(c1ccccc1Cl)C1CCC1 c1(CNC(c2nc(C(=O)OCC)sc2C)=O)cccc2scnc12.C12CN(C1)C2=O c1(C(C(=O)NCCNC(C2C(COC)C2)=O)C)ccc(Br)c(C)c1 N1(C(=O)NCC(c2ccc(F)cc2F)C)CCCN(C(F)F)CC1 CC(CC(=O)NCCCCNC(=O)CCn1cccc1)n1cc(Br)cn1 c1(C(=O)NC(C(C)NC(c2ccc(CC)o2)=O)C)cc(C)n(C)n1 c1(CCCC)ccc(S(=O)(=O)N2C(C(=O)NCC3(C)OCCO3)CC3CC23)cc1 CC1CN(C(c2cc(CC3CCC3)c[nH]2)=O)CC1Nc1ncc(I)cn1 C12(NC(C3CN(C(c4c(OC)n[nH]c4)=O)C(CO)C3)=O)CCC(CC1O)C2 C1(NC(C(F)=CC)=O)CN(C(C2CC(CC(F)(F)F)C2)=O)CC12CCC2 c1(CC)nc(C)[nH]c1C(=O)N(CCCN(C(=O)CCCNS(C)(=O)=O)C)C C1(CNC(c2scc(C)c2)=O)CC(C)N(C(=O)Cc2c(C(F)(F)F)coc2C)C1 N1(C(CSCCOC)=O)CC2CCC1C(NC(C1CC3CS(=O)(=O)CC3C1)=O)C2 CCCCC(O)C(=O)NCCC1CC(NC(c2cc3n(n2)CCC3)=O)C1 C(CCCCC(=O)NC1C=CC(CNC(c2cc(C(N)=O)c[nH]2)=O)C1)NC(C)=O C#CCC(C)(C)C(=O)N1CCOC(C(=O)N(C)Cc2cccs2)C1 C(=O)(C(CC(C)C)CC(C)C)N1CC2CCN(C(c3c(C)ccs3)=O)CC21 c1(C(=O)NCC(C2CCOC2)NC(C2(N(C)C)CCC2)=O)cc2scnc2[nH]1 c1(N2CCCC(CC)C2)nc(C)cc(=NC2COCC2OC)[nH]1 C=C1CON(C(=O)C(C2CCOC2)NC(=O)C(c2cccs2)SC)C1 CC1CCCC(C(N2CCN(C(=O)Nc3ccc(CCO)cc3)CC2)=O)C1 C(=O)(C#CC1CCCCC1)N1CC(C(C(=O)NCc2n[nH]cc2Cl)OC)C1 [N-]=[N+]=NCCCCCCC(=O)N1CCC2CN(C(=O)CCN3CCC(F)C3)CC12 C1(O)(CN(C(c2c(CC)nns2)=O)C)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C=C(C)C1CN(C(=O)NCc2nn(C)cc2C#N)CCO1 Cc1cnc(C(=O)NC2CC(C)N(C(C3(F)C(C)(C)C3(C)C)=O)C2)c(F)c1 C(C(F)(C(=O)O)C(C)C)COC(=O)NC(C(=O)NC)C(C)OC(C)(C)C N1(C(C#CCNC(c2cnc(OC)s2)=O)=O)CCC12CCCOCC2 c1(C(N2CC(NC(CC=CCC)=O)C3C2C3)=O)ccc(-c2ccco2)nc1O c1(C(=O)NCC2N(C(CCC(C)C)=O)CC(C)CC2)ccn2nncc2c1 Cc1cc(NC(=O)C(=O)N2CC(c3cccnc3O)C2)c(C)c(C)c1 N1(C(N)=O)CCC(C(N2CC3CC2C3NC(=O)C(=C2CCCCC2)F)=O)CC1 CC1CN(C(=O)CSc2cn[nH]c2)CCC1NC(c1ccc(CSC)o1)=O Cc1cc(C(=O)NCC2COCCN2C(=O)CC(C)C2CC2)nnc1O CC1CN(C(C23C(NC(=O)CNC(C4CC4C)=O)C4CC2C3C4)=O)c2ccccc21 c1(N(CCC)C)ccc(C(=O)N(C)CCN(C)C(C2CCC3CC3C2)=O)cc1 C1(NC(CC(C)OC)=O)CCC2(CC1)CN(C(=O)CCN(C)CCO)CCO2 CC1(C(=O)NC2CC(CNC(=O)CSc3ccc(O)cc3)C2)CCOCC1 C1(CC(=O)N(C(C)CO)C(C)C)CCCN(C(C(C)(C)C)=O)C1 CC1(C)CC(C)(CNC(c2cc(CO)[nH]n2)=O)CN1C(c1cccc[n+]1[O-])=O C1(C(=O)NCC(=O)Nc2ccccc2)CCC2CN(Cc3ccccc3)CC12 C(=O)(C(C(C)C)OC)N1C(C(=O)NCc2cc(COC)on2)CC1C c1(CNc2c(C)nn(CCC(=O)OC)c2C)cc(Cl)cc2c1CCC2 C1(C(C)=O)CC(CC(N2CCCC2(C)CNC(=O)CSc2nccn2C)=O)C1(C)C c1(C(N2CCC(C(=O)NCC3(OC)CCOC3)(CO)C2)=O)c[nH]c2ccccc12 C1(C2CC2)(C(=O)NC(CC#C)C(=O)NC)CN(C(c2nc[nH]n2)=O)C1 CC1CCCN(C(=O)Cc2c(F)cccc2F)C1CNC(C1(CCO)CC1)=O C1(NC(C(C)CC2CC2)=O)CN(C(c2ccccc2)=O)CC1O C(C(C)(C)C(C)(C)C)NC(C(Cn1cncn1)NC(COCCOCC#C)=O)=O C(=O)(CCCCCN(C(=O)C1=C(C)CC1)C)N(C1CCNC1=O)CC C(=O)(C#CC1(C)CCCO1)N(C(CNC(c1ccc(Cl)cn1)=O)C1CC1)C Cc1ccc(C(=O)NC2CCC(C)(CNC(c3onc(C)c3C)=O)C2)nc1C N1(C(c2cccc(CC)c2)=O)CCC(C(=O)NCCOCC(C)C)=C(F)C1 c1(C(N2CCC(CCC(=O)NCCOCCF)C2)=O)ccnc(O)c1 c1(OC)ccc(C(C(=O)NCC2CC2)N(C2CC(C)(C)C2)C)nc1C CC(C)(C#N)CC(=O)NCCC1CN(C(=O)C=Cc2cccc(CO)c2)CCO1 C1(C(C)C)CN(C(c2c[nH]c3cnccc23)=O)CCCN1C(=O)C=CC(=O)N(C)C Oc1cc(OCCCCCC2CCCNC2)cc(Br)c1.c12cccc(c1)S2 C1(c2onc(N3CCC(C)CC3)n2)CS(=O)(=O)CC1c1ccccc1 c1(C(N2CCCC(C(N3CCC4(CC3)N=N4)=O)CC2)=O)ccc2c(c1)CC2 C1(NC(C2CC2c2ccccc2)=O)CC(F)CN(C(C2CC3CCC2CC3)=O)C1 c1(C(=O)NCC(CO)NC(C2CC(C)(O)C2)=O)cc(C#N)cc2ccccc12 S(=O)(=O)(c1ccc2sc(Cl)cc2c1)NC1C(C)CCC1 C#Cc1cc(C(=O)NCCN(C(=O)C(C2CCCOC2)OCC)CC)ccc1C c1(C(=O)NCC2N(C(C3N(C)C(=O)CC3)=O)CC2)ccc(S(N)(=O)=O)cc1 c1(CC(=O)NC(C(=O)NC(CC)C2CC2)C2CCCC2)ccc(O)cn1 N1(CC(=O)NC2(CCCOC)CCCC2)CC(C)CCC1C C(C(C(F)(F)F)N1CCN(C(=O)C(C2CC2)SC)CC1)NC(C=C(CC)CC)=O Cc1ccc(S(=O)(=O)N2CCN(C3COCC3O)CC2)c(Cl)c1Cl C1(NC(CNC(CNC(C)=O)=O)=O)CCCN(C(c2n[nH]c(C)c2F)=O)CC1 c1(C(N(C2CCC(NC(CC(C)(C)OC)=O)CC2)C)=O)cnn2c(N)ccnc12 C1(C(=O)NCC(=O)NCCO)CC2CCCC2N1C(C1CCC(F)C1)=O c1(C(C(=O)OC(C(C(=O)OCC)=O)C)C)cc(C)cc(F)c1 c1(CC)cc(OC)ccc1N.C12(CCCCC1)C(=O)NCC(CO)CNC2=O c1(C(N(C2CCN(C(=O)CSC)C2)CCC)=O)ccc(OC)c(Br)c1 C1(N(C(c2ocnc2C)=O)CC)CCCN(C(=O)CCN2CCOCC2)CC1 N1(C(CC)=O)C2CCC1CC(N(C)C(C1CC(=O)N(C)C1)=O)C2 c1(C(=O)OC(C(=O)NCC)C)cccc2c1CCCC2 N1(C(CC(C)CF)=O)CC2CC1CCN2C(c1cnc2cc[nH]c2c1)=O CC1CN(CC2COC(C)C2)CCN1S(=O)(=O)Cc1ccc(F)c(F)c1 C#CC1(C(=O)NCC(O)C(C)(C)O)CCN(C(C2CC(C)N(C)C2)=O)C1 N1(C(C2NC(=O)C(F)C2)=O)CCN(C(C2(F)CC2)=O)CC1c1ccccc1 C1(C(=O)NCCC(C)N(C(=O)CC2CC=CCC2)C)CC2CC2C1 CCC(C(=O)N(CC(O)CNC(=O)CN(C)C)C)NC(N)=O N1(c2cc(N3CCC(OCC)C3)ncn2)CCC2(CCCOC2)CC1 c1(C(=O)NC2(CSC)CC2)sccc1CNC(C1CCCN1C1CC1)=O CC(C)C(O)C(C)C(=O)NCC1(CNC(c2ncc(F)cc2F)=O)CCCC1 N1(C(=O)NCC)CCC(c2nnnn2C2CC2)(NC2CC(=O)N(C)C2)CC1 N1(c2ccc(OC)cc2)CCC2C(CCCN2C(=O)OC(C)(C)C)C1 C(CC(C)(C)CC(=O)NC1(C(=O)NCc2noc(C(N)=O)n2)CCCC1C)OC n1(CCCC)nc(C)c(C(=O)NCC2CCCN2C(=O)C(CCO)N(C)C)c1Cl c1(C(N(C2CCN(C(c3cc(COC)[nH]n3)=O)CC2)CC)=O)nn(CC)nc1C C1(C(=O)NC(C)CC2CN(C(=O)CNC(c3ccoc3)=O)C2)CC(C2CC2)C1 C12=NNC(=NC3CC4CCC3N(C4)C1)O2.c1(CC)cnn(C)c1 C1(C)(C(N(CC(O)CNC(=O)CCNC(c2ccco2)=O)C)=O)CCCC1O CC(CC(=O)NC1(CNC(=O)CCC(=O)N(C)C)CCC1)P(C)(C)=O c1(CC(=O)N(C(CCNC(c2cc(C)ncc2)=O)C)C)ccc2cnccc2c1 c1(C(N2CC(CC(C)NC(C(C)NC(=O)NC)=O)C2)=O)ccccc1C1CC1 C1(C)(C(=O)NC2CCN(CCC)C2)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1 CC1CCCC(C(=O)N(C2CCCC2)CCCNC(C2(CO)COC2)=O)C1 N1(C(C)C2CC2)CC(C(=O)N(C)CCN(C)C(C2(C3CC3)CC2)=O)CC1=O N1(C(CCCN(C(CCC(C)N(C)C)=O)C)=O)CC(O)CC(C)(C)C1 c1(CC)c(C(=O)NCC(C)N(C(=O)C(C2CC2)SC)CC)nnn1COC c1(CN(C(C(C)N(C)C(C2CCCSC2)=O)=O)C)ccc(C#N)s1 N1(C(C(C)(C)NC(C(C)NC=O)=O)=O)CCCC(F)C1 c1(C(=O)NC2CC(NC(C(C)Cc3ccccc3Br)=O)C2)ccc(C#N)n1C N1(CC(=O)NCC2CC(F)(CNC(C(CC)N(C)C)=O)C2)OC(C)(C)CC1=O C1(n2cccc2)(CC(=O)NCC(C)CNC(=O)CN(C2CCCC2)C)CCCC1 N1(C(c2cc(C(C)C)on2)=O)CC(N(C)C(c2cnnc(O)c2)=O)C(C)(C)C1 CC(C(=O)NCC(C1CC1)N(C(=O)CCc1ccc(F)cc1F)C)C(C)(C)C C=Cc1ccc(C(N2CCOC(CNC(C3CCN(C)S3(=O)=O)=O)C2)=O)cc1 N1(C(c2cnn(C)c2C2CC2)=O)CC2CC1CCC2NC(c1ccoc1Cl)=O Cc1cc(=NC(=O)C(=O)NC2(C)CN(C(=O)CCc3ccc[nH]3)C2)[nH]o1 N1(C(c2cccc(C#C)c2)=O)CCC2CCN(C(=O)CC3CC34CC4)CC12 N1(C(C2CC3N(C(=O)OCC)C(CC3)C2)=O)CCc2ccc(O)cc21 c1(C(=O)NCc2nccc(C(=O)NC3CC34CCCC4)c2)c[nH]c2cnccc12 Cc1ccc(F)c(C(=O)NC2CN(C(c3cccc(CO)c3C)=O)CC2C)c1 Cc1ccc(CC(=O)NC2CCN(C(c3ccno3)=O)C2)cc1[N+](=O)[O-] C1(C(=O)NCC2CCC(NC(CSCCC(C)C)=O)C2)CC(C)(C)CCO1 n1(C2CCCC(C)C2)cc(C#CCNC(=O)C(C)(C)c2cnco2)nn1 CN(S(N)(=O)=O)CC(N1CC(C(N)=O)(CNC(=O)CCc2cncs2)C1)=O c1(C(=O)NCC(CNC(C=C(C)c2ccco2)=O)CO)ccc2c(c1)OCCN2 C1(C(C)C)CN(C(C2CCCN2C(=O)COc2ccc(Cl)cc2)=O)CCO1 C1(NC(CCc2cnc(C)o2)=O)CCN(C(c2nccnc2C)=O)CC1O C1(C(=O)NCCC2(O)CCN(C(CC3ON=C(C)C3)=O)C2)CC2CSCC(C1)C2 Cc1sc(Br)cc1C(=O)NCC1CN(C(C23CC(F)(C2)C3)=O)C2CC12 c1(CNC(c2cccc(Cl)c2Br)C)c(O)ccc(F)c1F c1(C(=O)NCCCN(C(C2CS(=O)(=O)C2)=O)CC)cc(C(F)(F)F)no1 Cc1nc(N(C(=O)CCC(F)(F)F)C2C3CNCC23)nc2ccccc12 C(CC(C(=O)N(C(C)CCNC(c1ccncn1)=O)C)OC)OC N1(C(C(C(CC)O)C)=O)C2CCCC1CN(C(C13CCC(OC)(CC1)CC3)=O)C2 C1(NC(C(C)COc2ccccc2)=O)CCCN(C(C2(O)CC(C)(C)C2)=O)C1 c1(C2CN2)ccc(CNC2CCOC2)cc1.OCCOCF c1(C2CCN(C(c3c(C)ccnc3)=O)CC2)nc2ccccc2[nH]1 Cc1ccc(F)cc1CC(N1CCC(NC(c2cnc(O)c(C)c2)=O)C(O)C1)=O Cc1cc(CC(N2CCC(CNC(c3sccc3Cl)=O)CC2)=O)cc(O)c1 N1(C(C(CN(C)C)(C)C)=O)CCC(C#N)(NC(=O)Cc2cc(F)ccc2F)C1 c1(C(N2CCCC(NC(c3cn(CC)nc3)=O)CC2)=O)ccc(F)c(C)c1Cl Cc1nsc(C(=O)N(CCCCN(C)C(c2sccc2F)=O)C)c1N C1(CNC(CNS(CC)(=O)=O)=O)CCC2CN(C(=O)CC3CCC(=O)N3C)CC12 c1(C(N2CCC(CNC(C(C3CCCCC3)C)=O)C2)=O)cc2cc(Cl)ccc2s1 C1(C)(C(N2CC(NC(Cc3ccc(C(C)=O)s3)=O)(CO)C2)=O)CCC(C)=C(C)C1 C1(NC(C(CC)CCOC)=O)CN(C(=O)CC2CCCC2)C2CCCC12 Cc1ccc(C(=O)N(CCCNC(=O)CC#N)CCO)c(-c2ccccc2)n1 N1(C(CC(CC=C)NC(c2ccc(C#N)c(C)n2)=O)=O)CC2CCCCCCC12 C(CNC(=O)CNS(C)(=O)=O)(CC(F)(F)F)NC(Cc1ccc(C)cc1)=O Cc1cc(F)ccc1C(O)C(=O)NCCN(C(C1CC1C1(C)COC1)=O)C1CC1 N1(C(c2c(CC)ncs2)=O)CC2CN(C(=O)Cc3cc(OC)no3)CCC12 C(C(O)C(=O)N(C1CCN(C(c2ccsc2C(F)F)=O)C1)CCO)SC C12(C(=O)OCC)CCCC1(CNC1CCC1CO)C2 C1(n2cnnn2)(C(=O)NCCN(C(C)C)C(C2CCN(C)CC2)=O)CCSCC1 c1(CC2(NC(CCc3cn(CC)nn3)=O)CCOC2)cc(C)cc(Br)c1 C=CCC(CC=C)C(=O)N(C(C)CNC(=O)C=C1CCC1)C N1(CC)CCC(C)(NC(=O)N(C(c2ccccc2)CO)C)C1 C=CCC(CC(=O)NC(C)(CO)C(F)F)NC(=O)COC1CCOC1 S(=O)(=O)(c1ccc(C)c(NC)c1)N1CCC(C(=O)NC2CC(=C)C2)C1 CCC(CCOC)C(=O)N1CCC(C(C)C(=O)NCC2(O)CSC2)C1 c1(C(=O)NC2CCC23CN(C(=O)CCc2cnc[nH]2)C3)c(O)nnc2c1CCC2 C1(OCC(=O)N(CCC)CCNC(C2CCC2C(F)(F)F)=O)CCCCC1 c1(C(=O)NCC(c2ccc(C)cc2C)OC)ccc(C#N)c(F)c1Br N1(C(CNC(CC(C)C)=O)=O)CCOCC(NC(c2ccsn2)=O)C1 C1(C(=O)NCCCc2cn(CC(CN(S(C)(=O)=O)C)(C)C)nn2)CC2C=CC1C2 CS(=O)CCC(=O)NCCC1CCCN(C(c2ccccc2OC2CCC2)=O)C1 C(=O)(C#CC1(C)CCCO1)NCC1(C)N(C(c2n(CC)ccc2)=O)CCC1 C(=O)(C(CO)C(F)(F)F)NC(C)C(C)C(=O)NCC1CC1c1ccoc1 C(CCN=C(NCC1CCC=CCC1)N1CCC(C(C)(C)C)C1)OCC c1(C(=O)NC2CCCC(NC(=O)CC3CCC(O)C3)C2)cc(F)cc(F)c1 C=CCCC(C(=O)NC1C(C)(C)C1(C)C)NC(C1CCN(C)C1=O)=O N1(C(CC2C(CC)C2)=O)CC(NC(c2cnn(CC)c2C2CC2)=O)CC(O)C1 C1(NC(=O)Cc2cccc(Cl)c2)C2CC3CN(C(c4c[nH]nc4F)=O)C1C3C2 n1(CC#C)ccnc1SCC(=O)NC1(C(=O)O)CCOC1 C12(C(N(CC(=O)OCC)C)=O)COCC1CN(C(C1CCCC3(CC3)C1)=O)C2 C(=O)(C(C(=O)NCc1cn(C(C)(C)CC(=O)OC)nn1)C1CCCC1)OCC CCC(CCCC(=O)NCCCCCSCC)NC(=O)CCc1ccccn1 C1(C(=O)Nc2ccc(CC)cc2)CCC2CCC1N2C(c1cccnc1NC)=O C(=O)(C(C)(C)C(=O)N(CCCCNC(=O)Cn1ccccc1=O)C)N(C)C c1(CC(=O)NC(C(C)NC(CS(=O)(=O)NC)=O)(C)C)cccc2ccccc12 C(c1ccc2c(c1)CCO2)=CC(=O)NC1C(C)CN(C(=O)CCC2CC2)CC1 c1(N(C)C)ccc(C(=O)NC2CC2C(=O)N(C2CC2)Cc2ccc(F)cc2)cc1 N1(C(CC=CCNC(c2ccc(C)c(F)c2)=O)=O)CCCNC(=O)C1C(C)C c1(C(=O)NC2(CNC(COCC#C)=O)CCOC2)cc2c(cnn2C)nc1O N1(C(CN(CC(C)C)C(=O)Cc2cnnn2C)=O)CCCCC1C c1(C(C)C)cc(N2CC3C(NC(C4(C(F)(F)F)CCCC4)=O)C3C2)ncn1 C(=O)(C1=CCCC(C)(C)C1)NC(CC=C)CNC(c1nc(CC)oc1C)=O Cc1nc(CNC(c2c[nH]c(=S)cn2)=O)oc1C(=O)NC(c1cnn[nH]1)(C)C C1(C(=O)NCCC(C)N(C(c2c(CCCC)ocn2)=O)C)CCS(=O)(=O)C1 CN1CCN(C(=O)CC2NC(=O)CNC2=O)CC1CNC(=O)Cc1csc(Cl)n1 N1(C(CCOC)=O)CCCC(C(N2CC(N3CC(F)C3)C2)=O)C1CO Cc1ccc(O)cc1CC(N1CCC(N(C(=O)Cc2ccccc2CO)C)C1)=O Cc1cc(C=CC(=O)NC2CN(C(c3ccon3)=O)C3(CCC3)C2)ccc1Br Cc1cc(NC(C2(CO)CC3CC3C2)=O)ccc1NC(=O)COC1CCC1 N1(C(C(c2c(C)nn(C)c2)C)=O)CC2CC(C)N(C(=O)COC(F)(F)F)C2C1 N1(C(CCCC2(NC(CCCCCSC)=O)CCC2)=O)CC(=O)N2CCCC2C1 Cc1nc(CC(C)C)oc1C(N1CC(C(C)NC(=O)Cc2csc(=N)[nH]2)C1)=O C(=O)(C(C)C(F)(F)C(F)F)NCCC1CCN(C(C(C(C)O)N(C)C)=O)C1 C1(C(=O)N)(CSC)CN(C(c2cnn(-c3ccccc3)c2)=O)C1.C1(S)CCCC1 C1(C(=O)NC(CSC)C(N2CCOC(C(C)O)C2)=O)CCN(C)CC1 c1(C(=O)NCCNC(c2ccc(C)c(Cl)c2N)=O)cc2sc3ccccc3c2s1 N1(C(CC(C=C)CC)=O)CCCCCC(NC(c2ccc(C#N)n2C)=O)C1 CC(F)(F)C(C)(C)CC(=O)NCC1CCN1C(=O)Cc1cnn2ccccc12 N1(CCC(=O)N(CCN(C(=O)CC(=O)NC2CC2)C(C)C)C)CCCCC1=O CC1CC(F)(F)CCN1C(C1N(C(c2cscc2Cl)=O)CC12CCCC2)=O CCCC(CCCNC(c1ccon1)=O)NC(=O)C(C(C)(C)C)c1ccccc1 C1(C)(CNC(C2CC(OCC)C2)=O)CN(C(C2(CC(C)C)COC2)=O)CCO1 CC1(NC(C2CC(n3cnnc3)C2)=O)CCCN(C(C2(SC3CC3)CCC2)=O)C1 Cc1cccc(C)c1OCC(=O)NCC1(CNC(C2CC23CC(O)C3)=O)CCC1 N1(C(c2nn(C)c(Cl)c2)=O)CCC2CN(C(=O)C(F)C3CCCC3)C2C1 N1(CC)CC(NC(c2occc2CNC(c2coc(C(C)C)n2)=O)=O)CCC1=O c1(C(N2CCCC2)=O)cc(Cl)cn1C.CCC1CNC(=O)C2CC(C2)CN1 C(=O)(C1=C(Cl)CCOC1)N1CCC(O)(C(CNC(c2c(C)csc2)=O)C)C1 C1(OC)CCC2(C(=O)Nc3cccc(NC(=O)C(C)OC(C)(C)C)c3)CC12 CC1(C)CC(NC(c2cncc(O)c2Cl)=O)CCN(C(=O)CCCCC2CC2)C1 N(S(=O)(=O)N(C)C)CC(N1CC(O)(C(C)NC(=O)C=CSc2nc[nH]n2)C1)=O c1(OC)cc(Nc2ccccc2)nn1C.c12cscc1C(=O)N2 Cc1ccc(CN2CCC(C)C2c2cn(CCc3ccccc3)nn2)nc1F N1(C(C2N(CCC)CCC2)=O)CC2CCC(C1)C(NC(C1CNC(=O)N1)=O)C2 c1(NC(C2C(C(=O)NCc3ccc(OC)nc3)C2)=O)ccc(F)nc1C Cc1cc(CNC2CCN(CC(F)(F)F)C2)c(C)[nH]1 N1(C(C=COCC)=O)C2CCC1C(CNC(c1ccc(=N)[nH]c1Cl)=O)C2 CC(C1CCCCC1)=CC(=O)NC1COC2(CNC(=O)Cn3cccn3)CC1C2 C(C(=O)Nc1cc(C)ccc1O)(C(C)CC)NC(CC=CCC)=O C(=O)(C(C)(C)C(C)(C)O)N(C1CCN(C(c2cnc(C(C)OCC)s2)=O)C1)CC c1(NC(c2nc(CC)[nH]n2)C)nccc(=NC(C)c2nccn2C)[nH]1 C1(NC(C)=O)CCN(C(=O)C(O)CC2CC2)C(C)C1.N12CCCC1SCC2=O C1(C(=O)NC(C2CCCN2C(c2ccc(SC(F)(F)F)o2)=O)(C)C)CCCCS1 C1(C(=O)OC)CC(C)N1C(=O)C(CC1CC1)NC(=O)CCOCC(C)(C)C Cc1cccc(C(N2CCC(NC(=O)CC3CCCC34CC4)C(F)C2)=O)c1C c1(C(N(CC(C)CO)C)=O)cc2c(s1)CCC(C(C)(C)C)C2 c1(OC)nc(C)c(Br)cc1CNc1cncc(Cl)c1 CC(F)(F)CCC(=O)NC1CC2CC1N(C(C1CCCC1(C)C)=O)C2 C1(CNC(=O)C(F)F)CC=CC(n2cc(COCCO)nn2)C1 N1(C(c2cc(C)on2)=O)CCCOC(CNC(=O)CC(C(F)F)c2ccccc2)C1 C(C(C(=O)N1CC(OC(=N)O)C1)C(C)(C)C)NC(C1(CC=C)CC=CC1)=O C(=O)(C(C)(C)CS(C)(=O)=O)NC(CCNC(CCC(CC)C)=O)Cc1ccccc1 C(=O)(C(C)(C)C(=O)NC)NC1CC(NC(c2c(C#C)c[nH]n2)=O)C1 CC(CN=c1ccnc(NC2COC3(CCC3)C2)[nH]1)C1CCC1 CN1CCC(C(=O)NC2CC(CO)N(C(C34CC(C#N)(C3)C4)=O)C2)C1=O N1(C(C=CCC)=O)CCCC(C)(CNC(c2c(OC)ncnc2C)=O)C1 c1(OC)c(C(=O)NC(C2CN(C(c3cc(O)cs3)=O)CCO2)C)c(C)nn1C CC#CCCCC(=O)N(C(CC(C)C)C(=O)NCc1ccc(OC)cn1)C CC1CCC(C)CN1C(C1CN(C(=O)C(CCC=O)=CCN)CC12CC2)=O N1(C(c2c(C)onc2C2CC2)=O)CCOC2(CCN(C(c3cocn3)=O)C2)C1 c1(C(N2CC(C)(NC(c3c(CC)scc3)=O)C2)=O)cn(CCOC)nc1C c1(C(=O)NC2CN(C(C(CCC)OCC)=O)CC2O)ccc2nnnn2c1 C1(C(=O)NC2CCCN(C(C3CCC(O)C3)=O)C2)CCn2nnnc2C1 C1(NC(=O)C=Cc2cncs2)CN(C(c2ccc(-c3csnn3)cc2)=O)CC1F Cc1cccc(NC(=O)NCCC(=O)N(C)CCNCCC(C)(C)N)c1C CCC(C(=O)N1CC2CC2(CNC(c2cc(CN(C)C)c[nH]2)=O)C1)C(C)C C1(N(C)CC#N)CCN(C(=O)CCCc2cnn[nH]2)CC1O C(=O)(CS(=O)(=O)CC(C)C)N(C1CCN(C(C2(C)CCOC2C)=O)C1)CC C(C)(C)(CN=c1[nH]c2c(c(=NC3CCCN(CCOC4CC4)C3)[nH]1)CCC2)NCC Cc1nc(C(=O)NCC2CC3CC3N2C(C2CN(C3CCC3)C2)=O)cn1C(F)F C(=O)(CCC(CC)NC(C1(CC(C)C)CCC1)=O)N1CCC(CC#C)CC1 N1(C(CCSCCCC)=O)CC(NC(=O)CC(C)C(C)C)C(C)(C)C1 c1(C(=O)NC2CN(C(C3CCc4n[nH]cc4C3)=O)C2)c(F)ccc2nc[nH]c12 C1(NC(C(CC)C)=O)CN(C(=O)CCC(=O)c2ccncc2)CC1N=[N+]=[N-] CON(C)C(=O)C(CC(C)C)NC(c1cncc(CO)c1)=O C12(CC(=O)NCC(=O)NCC(C)C3CC3)CCC(CC1)N2C(=O)CN.C(C)(C)(C)N C1(O)(CC(=O)Nc2cnn(C3CC3)c2)CCCOC1.CC1(C)C2C1CNC2=O c1(C(C(=O)NCc2nccc(N)n2)F)c(F)cccc1F C1(OC)(CNC(C2SCCCS2)=O)CCN(C(c2csc(Cl)n2)=O)C1 c1(C(=O)NCC2(C)N(C(CCOC)=O)CC(F)(F)C2)ccc2c(c1)CCCS2 c1(SCC(=O)NCCOC)ncc(C(N2CC(NC(=O)CC(C)C)C2)=O)cn1 c1(CC(=O)NCC(CNC(CC2(COC)CC2)=O)F)cccc(C(F)(F)F)c1 C(=O)(CC(C)(C)CCC)NC(CNC(C(CC#C)C)=O)C C(=O)(NNC(=O)c1ccc(OCc2cscn2)cc1)C1CCC(=O)N1 CC(C(=O)NCC=CCNC(c1ncccc1OC(F)F)=O)C(C)C(C)(C)C CC1=NNC(=O)C1CC(=O)N(CCC(=O)NCc1nn[nH]c1C1CC1)CCO C#CC1CCC1C(=O)NC1COCC1NC(=O)CC(=O)OC(C)(C)C C12(CSC3CCCC13)c1nnnn1CCN2CCF.C1(SCC)CC1 N1(C(C23CCC(CN(C(CC4CC(SC)C4)=O)C2)C3)=O)CCc2nn(C)cc2C1 c1(CC)ccccc1OCCC(=O)NC(C)COC(O)CN(C)C N1(C(C2COCCN2Cc2c(F)cccc2Cl)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(CN2CC3C(C(N4CCCN(CC)CC4)=O)(C3)C2)ccc2ccc(Br)cc2c1 N1(C(c2nc(C)sc2C)=O)CCC2(CC1)CC2(CO)CNC(C1CCC(=O)N1)=O O(NC(=O)CCc1cn(C)nn1)CC(C)O c1(C(N2CCC3(NC(c4ccc(Cl)cc4Cl)=O)C(C2)C3)=O)ccnc2[nH]cnc12 CC(C)(CCCC(=O)N1CCC(O)(C(N)=O)C1)NC(c1sccc1CO)=O c1(OC)ccc(NC(=O)CC2CC2CNC(=O)CC2CC(F)C2)cc1O c1(OCCN2CCN(CC3C(CC)C3)CC2)cccc([N+](=O)[O-])c1 N1(C(CC2(C=C)CCCCC2)=O)CCN(C(C2CC(=O)N(OC)C2)=O)CC(C)C1 C1(OC)CCCN(C(=O)CC2(C)CCN2C(=O)CN2CCCCC2C)C1 Cc1ccc2nc(C(N3CC4(CCCCN4C(=O)C#CC4CC4)C3)=O)c(N)n2c1 C1(C(=O)NC2C(C)(C)CN(C(=O)COC3CC3)CC2)CCS(=O)(=O)C12CCC2 Cc1cc(C(=O)N(C)CC2CCCN2C(c2cscn2)=O)nn1C(C)C1CC1 N1(C(C2CCCC(NC(c3ccc(Cl)c(F)c3)C)C2)=O)CCN(C)C(=O)C1C N1(C(c2cccc(OC)c2F)=O)CC2CN(C(=O)Cc3nc[nH]n3)CC2C1 C(=O)(CCC1=NNC(=O)CC1)N(C1CCCCC1)CCNC(C1C(C)(C)C1)=O C1(NC(C=C(C)Cl)=O)CCN(C(=O)Cc2cn3cc(C)sc3n2)CCC1CO CCC(C)C(C(=O)N1CCC(=CC(=O)NCc2cc(C)ccc2F)CC1)N(C)C C1(NC(c2cc(C)[nH]c2)=O)CCCC12CCN(C(c1conc1C(C)C)=O)CC2 c1(C(N(CCNC(c2cnn(C)n2)=O)CC)=O)c(C)nn2c(C)cc(C)nc12 c1(C(N2C(COC)CCC2)=O)c(-c2cnc(F)cc2F)cncc1F c1(CC(=O)NC(C)(CNC(=O)C(F)CC2CC2)C2CC2)ccc(F)c(Cl)c1 C1(CC(=O)OC)CN(C(=O)C(=O)NC2CCCNCC2)CCO1 C1(N(CCC)C(c2cc(Cl)cs2)=O)CCN(C(C2CCS(=O)CC2)=O)CC1 C=CCC(CC)C(=O)NC1(CNC(=O)C(C)NC(c2cccc(C)c2)=O)CC1 N1(CCCNN2CCCC2)CCCC(N=c2nc(SC)c3c(ncn3CC)[nH]2)C1 N1(C(c2c(C)cn(C)c2)=O)CCC(O)C(N(C(=O)CCOCCN(C)C)C)C1 Cn1cc(S(N)(=O)=O)cc1CC(=O)NCCCNC(=O)CCc1ncc[nH]1 c1(CCNC(c2n(CC)nnn2)C2CC2(C)C)ccc(-c2cccnc2)c(F)c1 C1(NC(c2n(C)nnc2)=O)CCN(C(C2OCC3CCCC2C3)=O)CCC1(F)F C1(CC)(NC(C2CCCC2C)=O)CCN(C(c2ccn(C(F)F)n2)=O)CC1 C1(C(=O)N(C(C)CN2CCCC2)C2CC2)C2CC3C(C2NC(=O)CC2(C#N)CC2)C13 c1(C(N2CCN(C(C3C(C(N)=O)C3)=O)CC2CC2CC2)=O)ccnc2[nH]cnc12 c1(C(N2CCC(CN(C(C3C(C=C)CC3)=O)C)C2)=O)cc(O)nc2c1CCCC2 C1(NC(C2(C)CN(S(C)(=O)=O)C2)=O)CCN(c2nccc(N3CCOCC3)n2)CC1 C1(NC(c2nc(OCC)oc2)=O)CC2CC(NC(c3csc4nnsc34)=O)CC12 O=C(C(CC(F)(F)F)c1ccccc1)Nc1cc(F)cc(C(=O)O)c1O N1(C(c2cnc(C)n2C)=O)CC2(CCNC(C3(C)CC3(C)C)=O)CCC1CC2 c1(C(=O)OC)c(C)nc2c(NC(C3CC(=O)CC(C)C3)=O)cccn12 c1(C(=O)NCCC(C)NC(C2CCOC2c2ccncc2)=O)cc(N)cc(F)c1 N1(C(c2c(C)oc(Cl)n2)=O)CC(C2CN(C(=O)C=Cc3ccc(C#N)cc3)C2)C1 C1(NC(C(=O)Nc2ccc(Cl)c(F)c2F)=O)CCCC2(C1)CC2(F)F C#CC1CCCN1C(c1cccc(-c2cccc(F)c2)c1)C(=O)NC c1(C(N2CC3C(C(=O)NC)(CC3)C2)C(=O)NC(C)C)ccc(OC)c(F)c1F c1(C(=O)NC(C2CN(C(C3CCSCC3)=O)C2)C)cccc(C(F)(F)F)c1 c1(OC)cccc(C(N2CCN(CC(C)O)C(C(C)C)C2)C(=O)OC)c1Br C(=O)(C(C)(F)C(=O)NCCOCCNC(=O)C(C)OCC1CC1)OC Cc1occc1CNCCCNC(=O)Cc1coc(C(F)F)n1 C1(NC(C2CC(OC)C2)=O)CC(NC(c2sc(N(C)C)nc2C)=O)C12CCC2 N1(CC)CC(C(=O)N2CC(C)(NC(=O)CC3=CCCCC3)C2)c2ccccc21 CCC(C)(CC)C(=O)N1CC(NC(=O)CC2SC(=N)NC2=O)C(n2cccn2)C1 C1(NC(C(CC=CCC)C)=O)CCN(C(=O)CC2(NC(C)=O)CC2)C(C)C1 CCC1=C(C(=O)NCC(C)NC(C2CC2c2c(F)cccc2Br)=O)CCCO1 N1(C(c2c(C)nns2)=O)CC2(C(N3CC(F)(F)CCC3C)=O)CCC1CC2 C(=O)(C1=CS(=O)(=O)CCC1)N(CC(C)O)CCNC(=O)C=CC1CCCC1 C12(C(=O)Nc3ccc(C)cc3F)CCC(CC1)N(C(c1cc3occc3[nH]1)=O)C2 Cc1ccc(NC(C23CC2CN(C(c2ccc(Br)cn2)=O)C3)=O)c(I)n1 C(=O)(C1=CS(=O)CCC1)NC(C(C)C)CCNC(c1ncccc1O)=O C(C(C)S(N)(=O)=O)NC(CCN(C(=O)CCOCCCOC)CC=C)=O N1(C(C(C)(F)F)=O)CCCCCC1CNC(=O)CC1CC2(CC2)C1 C1(NC(Cn2nc(C)c(Cl)c2)=O)CC(CNC(=O)CN(C)C2CC2)C12CCC2 Cc1noc(C)c1C=CC(=O)NCC1CCCC1NC(=O)CCc1cnn(C)n1 N1(C(C#CC(C)C)=O)CC2CC1CN(C(c1cccc(F)c1Br)=O)C2 C(C)(C)(CC(=O)N1CC(F)CC1CNC(=O)CCCc1csc(=N)[nH]1)SC N1(C(CCC(C)C)=O)CCN(C(=O)CSc2ccccn2)CC1C(C)C C1(NC(CC2C(C)CC=CC2)=O)CC12CCN(C(c1cc(N(C)C)ccc1F)=O)C2 c1(C(=O)NCC(CNC(c2c(C)cc(Cl)cc2)=O)C)cc(O)c2ccsc2c1 c1(C(N2CCC(C(C(=O)NCCC(CCC)C)(C)C)C2)=O)ccc(C)c(F)c1 c1(C(=O)NC)ccc(C=CC(=O)NC2CCCC2NC(C2CCC2C)=O)cc1 N1(C(c2c(C)csc2)=O)CCCN(C(c2coc(Cn3cccn3)c2)=O)CC1 C1(CC)CN(C(c2cnc(O)c(F)c2)=O)CCN1C(=O)CCN1CCCS1(=O)=O C1(c2cn(CC(=C)CC)nn2)CCCCN1C(c1cccc(OC)n1)=O c1(C(N2CCCN(C(=O)C(F)C3CCC3)C(CO)C2)=O)cc2c(nn1)CCOC2 C1(F)(C(N2CC(O)(CNC(=O)CC3CCCNS3(=O)=O)C2)=O)CCS(=O)(=O)C1 C1(NC(CCc2cc(C)[nH]n2)=O)CCC(C)(NC(C2CC(C3CC3)=NO2)=O)CC1 c1(CCCC(=O)NC2CC(n3cc(CCOC)nn3)C2)ccc(Br)cn1 c1(CC)n[nH]cc1C(=O)NCCCCNC(c1n[nH]cc1Cl)=O N1(C(=O)COCCNC(CSC)=O)CCN(C(C2COCCC2C)=O)CC1 C12(C(=O)NCC(C)(C)CNC(=O)C3CC3)CCCN(CCC1)C2 N1(C(c2cc(OC)no2)=O)CCCN(C(=O)CSc2ccc(C)s2)CC1CO N1(C(Cc2ccc(SC)cc2)=O)CC2(CCCN2C(=O)CSc2ccccc2)C1 C1(C(C)C)C(NC(=O)CCn2ncn(C)c2=O)CCN1C(c1ccnn1CF)=O C1(CNC(=O)C2=CCCOC2)CC12CCN(C(=O)C(O)CN1CCCC1)CC2 C12(CNC(CCCNC(=O)OCC)=O)CC1CN(C(=O)Cn1cccnc1=O)C2 Cc1cnncc1C(=O)NCc1ccnc(C(=O)NCc2nnc(O)n2C)c1 c1(C(=O)NCCC(C)(C)NC(c2c(C)nc(C)[nH]2)=O)ccc2sc(O)nc2c1 N1(C(=O)CCC2CCOCC2)CC2(CCCCN2C(=O)CC2(C(F)F)CC2)C1 c1(C(N2CCN(C(c3c(C(C)C)ncs3)=O)CC2)=O)cc(Cl)cc(C(F)(F)F)n1 c1(C2C(C(N3C(C(=O)NCC#C)CCC3)=O)C2)ccccc1C C(=O)(C(CCC)=Cc1ccccc1)NCC(CC)NC(c1ccoc1C(C)C)=O C1(C)(C(N(C(C)CNC(=O)CC2CCC3CC23)CC)=O)CCC(=O)C1 CC1CN(C(=O)CCCC(N)=O)CCC1CNC(=O)C=C1CCSCC1 N1(C(C(C2CCOC2)OC)=O)C2CCC1CN(C(=O)C1=C(Cl)CC1)CC2 C1(C(N(CCCN(C(C2C(C)=C2)=O)C)C)=O)(NC(N)=O)CCC1 c1(NC2(c3n(C)cnc3)CCOC2)nc(N2CCOC(C3CC3)C2)nc2sccc12 c1(COCC(CN(C2CCOC2C)CCCC)O)ccc(Cl)cc1 N1(C(c2cnn(C)c2Cl)=O)CCC2(NC(=O)Cc3cccc(F)c3)CC2C1 c1(OC)ccc(OC)c(CCN(C)CC(C(=O)OC)C(C)Cc2nnn(C)n2)c1 C1(CNC(c2nc(CS(C)(=O)=O)oc2)=O)CC2(CCC2)CN1C(C1CC1CF)=O CC1CCC(NC(c2ccc(OCF)cc2)=O)CN1C(=O)CC1CC2(CC2)C1 C=C1CC2(C1)CC(C(=O)NCC(O)CNC(=O)CCCSC(C)(C)C)C2 N1(C(C(c2ccccc2)C)=O)CC(CNC(=O)CCC2CC(F)(F)C2)C2(CC2)C1 CC(C)C(=O)C(=O)NC(C1(C(=O)N(C2CCCC(O)C2)C)CC1)C c1(OCC)cc(CN2CCN(C(c3ccno3)=O)CC2C(F)(F)F)ccc1C C(=O)(C(C#N)C(C)C)N1CCC(CC2N(C(C=C(CC)C)=O)CCOC2)CC1 C1(NC(C(C)Cc2cccc(Cl)c2)=O)CCN(C(=O)CCCCC#N)CC1C CCCCCCCCC(F)C(=O)NCC(O)CCNC(c1c(C)nsc1N)=O c1(C(N(C(CC)CO)CC2CCC2)=O)noc2c1COCC2 CC(CSCc1ccccc1)C(=O)NCC(C)(C)CC1CN(C(=O)CNC(N)=O)C1 c1(C(=O)NCC2CCN(C(C3CN(C(N)=O)C3)=O)C2)cnc2sccn12 c1(OC)nccnc1C(=O)NCC1CCCN1C(C1CC(=O)N(C)C1)=O c1(C(=O)NCCC(CNC(C(C)OC2CCOC2)=O)O)ccc2c(c1)CC(=O)N2 C1(NC(=O)NCCC2CC(O)C2)CCOCC1 Cc1cccc(S(=O)(=O)CCCN2CCCC(N(C)Cc3cn(C)nc3C)C2)c1 CCCC(CC(C)C)C(=O)N1CC(OCC(=O)NC(CC2CC2)CC)C1 C(=O)(CC(C)CNC(C1CC2CCC1C2)=O)N(CCC#C)CC CC1(C)OCc2cnc(NCC3CCC4(C3)OCCO4)nc21 Cc1ccc(=O)n(CC(=O)NC2CC2CNC(=O)C=CC(C)C)n1 C1(C(=O)NCC23CC(NC(C4CCN(CC)C4)=O)(C2)C3)CCC(F)(F)CC1 c1(C(N(C2(CC=O)CC2)C)=O)c(C)nn(C)c1N.c1(C(C)OC)ncc(F)cn1 CCCC(C)(CCC)C(=O)NCC1(NC(=O)C=Cc2ncccc2C)CCOC1 c1(-c2nnc(NC(CC(C)C3CC3)=O)o2)cccc(F)c1 C1(C(=O)NC(C2(CNC(CCOCCCCC)=O)CC2)C)CC(=O)NC1(C)C c1(OC)ncc(C)cc1C(=O)NCC(O)CNC(c1ccc(N)c(Cl)n1)=O c1(C(=O)NCC(CCOC)NC(C2CCCC2C(C)C)=O)cccc(OC)c1 C(=O)(C1=NN2CCCN=C2N1)N(C(CNC(C1(C(C)C)CCCO1)=O)C)C C(=O)(CS(=O)(=O)c1ccccc1C)N1CC(N(C)C(c2cc(N)cc(O)n2)=O)C1 CC1CN(C(c2ccn(C)n2)=O)CC(C)N(C(c2ccc(Br)cc2N)=O)C1 N1(C(C(C)OCC=C)=O)CC(C)(C)CC1CNC(C1(C(=O)OCC)CCC1)=O.CCCO N1(C(Cc2cc(C)[nH]n2)=O)CCC(N(C(=O)CCc2ccccc2Cl)C)C(C)C1 CCCC(O)CC(=O)NC12COC(CNC(=O)C(C)C3CCCO3)(C1)C2 Cc1cc(C)n2ncc(C(N3CCC(C4(NC(=O)C(O)C(F)F)CC4)C3)=O)c2n1 C#CC1CN(C(=O)C(c2ccco2)NC(C2CCCC3(CC3)C2)=O)CCO1 C(=O)(C(F)(F)C1(O)CCC1)NCC(C)(C1CC1)NC(c1ccc(C(F)(F)F)s1)=O C1(CNC(c2c(CCC)n[nH]c2)=O)COC(C)(C)CN1C(=O)CCC(C)N(C)C CC1CC(NC(c2ccon2)=O)CCN1CC1CCCS(=O)(=O)C1 C1(C(N2C(CNC(C3C(COC)C3)=O)CCC2)=O)C2CCC(CC2)C1C(F)(F)F Cc1ccc2c(c1)C=C(C(=O)NC1CC(N(C)C(C3CCCC3(F)F)=O)C1)CO2 Cc1cccc(C(=O)NC23CC(C2)N(C(C2(c4nccs4)CC2)=O)C3)c1 n1(CCC)cc(C(=O)NC2CCCC2CNC(=O)CCCc2ncc(C)o2)cn1 N1(C(CC(C(=C)C)O)=O)CCC2(CC1)CC(C)N(C(c1ocnc1C)=O)C2 C12(C(N3CC(NC(c4nccc(CC)c4)=O)C(O)C3)=O)CCCN(CCC1)C2 c1(OCC)cncc(C(=O)NC2CN(C(c3cn(CC4CC4)nn3)=O)CC2C)c1 C1(CN(C(=O)C(N2CCCC2)C2CC2)C)CCN(C(=O)CCc2cscn2)CC1 C(CC(C)(C)CC(=O)N(C1CCN(C(c2sccc2C(C)C)=O)CC1C)C)OC c1(C(=O)NC2CCN(C(C(=O)NCCCC)C)CC2C)cccc2nn[nH]c12 N1(C(C=C(C)Cl)=O)C2CCC1CC(NC(c1n[nH]c3c1CC1CC31)=O)C2 n1(CC(=O)NC2CC(CNC(C3CCO3)=O)C2)ccc(Br)cc1=O O=C(C1=CCCCO1)C(CCN(C1C=CCC1)CCO)=O.N C1(CC=C)(NC(=O)C=CCN(C(=O)CCC=CC(C)C)C)CCOC1 C(=O)(C(F)CC(C)(C)C)NCC1(NC(c2scc(C)c2)=O)CCCCC1C C12(C(=O)NC3C4CCN(C(CN(C)C)=O)C4C3)CCCC(=O)N1CCC2 c1(CN(CC#C)C(C2CC(=O)N(c3ccc(C)cc3)C2)=O)cccc(Br)c1Cl Cc1nn(C)c(C)c1C(C)NC(=O)C(=O)NC1CCCCC1F C(=O)(C(CCS(C)=O)N(C)C)NCC1CCC(NC(CCCNC(C)=O)=O)C1 c1(CC(=O)NC2(CC(=O)N(CCCN(C)C)C)CCC2)ccc(Cl)s1 C1(C(=O)NCC2CN(C(N)=O)C2)(OC)CCN(C(=O)Cc2ncc(C)s2)C1 N1(C(CCN(CC)CC)=O)CC(C)(C)C1C1CCN(C(=O)C(C)NC(N)=O)CC1 c1(C(N2CC(NC(CCCOC(C)C)=O)C3C2C3)=O)cc2c(nc1O)CCOC2 N(C(=NCCc1ccccc1)NCC1C=CCC1)CC(C)(C)N1CC1 C12(NC(C(C)OCC)=O)CC(C1)N(C(C1CCCOC1c1ccc(C)cc1)=O)C2 C1(NC(c2ccc3cccnn23)=O)CC2CC(C1)N(C(=O)C=C1CCCC1)C2 c1(CN(C(=O)NC2C(OCC)COCC2)C2CC2)ccc(Cl)c(Cl)c1 N#Cc1ccccc1C(=O)NCC1(NC(=O)CCc2ccccc2)CC1 C=C=CCCC(=O)NC1CC(F)(CNC(=O)CCC(=O)OC2CCCC2)C1 c1(C(N2CCN(C(C3CCCC(OC)C3)=O)CC2CF)=O)coc2c1CCCC2 C1(CNC(CSCCC(C)C)=O)C2CN(C(C3CC3C(N)=O)=O)CC12 c1(CC(=O)NCc2ccccn2)cc(Br)ccc1Cl C(CC)(CC(F)(F)F)NC(C1C(NC(C(C(C)C)OCC)=O)CC1)=O C1(CC)(CNC(c2nnnn2CCOC)C2CCC2)CCCC1 C(=O)N=c1nc[nH]n2cccc12.CC(C)CC(O)C(=O)N(C1C(N)CCCC1)C C1(C(=O)NCC2CCCN(C(C3(OC)CC(C)C3)=O)C2)CN2CCN1CC2 c1(C(N(C2CCN(C(=O)C(n3cc(Cl)cn3)C)C2)CC)=O)cc(C)cc(C)n1 c1(CC)c(C(=O)N(C2CCN(C(=O)CCSc3nccn3C)C2)CC)ccn1C c1(NC2(C3CN(C(C(C)O)=O)C3)CC2)ncnc2ccc([N+](=O)[O-])cc12 Cc1c(C(=O)NCC(C2CC2)NC(c2cnn(C)c2Cl)=O)[nH]c2cc(F)ccc12 c1(C(N2CCC(NC(COCCC)=O)(CF)C2)=O)cnn2cccnc12 CC1(NC(C2(c3ccccc3)CC2(C)C)=O)CCN(C(=O)CS(N)(=O)=O)CC1 Cn1ccc2cc(C(=O)NC3CC(O)CN(C(=O)CSC(F)F)C3)cnc12 CCC(C)(C)C(O)C(=O)N1CCCCC1CC(=O)NCC1CC2CCC1O2 CCCCC(C)(C)NC(=O)C(C)C(C)NC(=O)CC1CCOC1 c1(OC)cnc(C(N2CCC(CCNC(c3cc(C)n(C4CC4)n3)=O)C2)=O)cn1 c1(C(=O)NC(CC)CN(C)C(C2(N=[N+]=[N-])CC2)=O)cc(C)nn1C1CC1 C1(C(=O)OC)CN(C(C2CCOC(C)(C)C2)=O)C2(CCC2)C1.c1cn(C2CC2)nn1 C1(C)(CNC(C(C(C)C)O)=O)CN(C(=O)C(C)(C)C2CC2)CCO1 C1(NC(=O)Cc2cnns2)CC2CCCC(C1)N2C(C1(CF)CCC1)=O C1(C(=O)NCc2ccc(CO)o2)CCCCN1C(c1cnc(O)[nH]1)=O c1(C(CNC(c2ccc(C(O)C(F)(F)F)cc2)=O)=O)ccc(F)c(Cl)c1 c1(C(N2CC3(CC3C(N3CC4CC4C3)=O)C2)=O)cccc(Br)c1F Cc1ccc(C(=O)NC2CCN(C(=O)CC3CSC3)C(C)C2)c(Br)c1F C1(CNC(CC=C)=O)CCC2(CCC2)C1NC(=O)CC#CC C1(NC(C(N2C(=O)CCC2=O)C)=O)COCCC1N(C(C1CCC(C)CC1)=O)CC Cc1ccc(C(=O)NC2C3CC2N(C(=O)CC2CCC4CC24)C3)cc1S(C)(=O)=O S(=O)(=O)(c1ccc(=NCCc2ccc(F)cc2F)[nH]c1)NCC(=O)NCC1CC1 CC(C(=O)NC1CCOCC1NC(c1c(Cl)nn(C)c1Cl)=O)C(C)(C)C CC1(C)OCC2CC12C(N1CCC(C)(CNC(c2nccc(Cl)c2O)=O)C1)=O CC(CNC(=O)C(c1ccn(C)n1)C)CC(=O)NC(c1nc[nH]n1)CO c1(C(=O)NCC2CN(C(c3ccc(Cl)o3)=O)C2)cc2ccc(F)cc2[nH]1 c1(C2C(C(N(C(C)CNC(=O)C(CO)c3ccccc3)C)=O)C2)ccc(Cl)nc1 Cc1cccc(Br)c1C(C(N1CCC(N(C)C)CC1)=O)NC(C1CC1F)=O N1(C(c2c(C)nc(O)[nH]2)=O)C(C)CC2CN(C(=O)CNC(=O)OC(C)(C)C)CC12 C1(C)(COC)CC(NC(c2ncc(F)cn2)=O)CN1C(c1c[nH]nc1OC)=O CC(C(C)C(=O)NC(C)(C)C(=O)NO)NC(=O)Cc1cn(C)cn1 C1(NC(c2[nH]ccc(=N)n2)=O)CC12CCC(NC(=O)CC1COCCO1)CC2 c1(C(C)C)ccc(C(N2CC3CN(C(=O)C(C)Cc4ccco4)C3C2)=O)cc1F CC(C)(C(=O)NCc1cc(C(=O)NCC2(F)CC(O)C2)no1)C1CCC1 CCCC(O)C(CO)NC(C1CCC2(CC2)N1C(C1CC1(Cl)Cl)=O)=O c1(C(=O)NC2(C3N(C(C4C(=C)CC4)=O)CCC3)CC2)n[nH]c(C)c1Cl N1(C(=O)CCc2ccncc2)CCC2(CCCCN(C(=O)C3=CCCC3)C2)C1 N1(C(CCCOCC=C)=O)CCOCC(NC(C2COC(C)(C)CO2)=O)C1 CC1CC(NC(c2cccc(CCO)c2)=O)CN(Cc2ccsc2)C1 C(=O)(C#CC1CCCOC1)NC(C1CCN(C(=O)C(C)(F)F)C1)C C(CC(C)(C)C)(C(=O)NC1CCOCC1C(=O)NCCOCC(N)=O)OC c1(C(N(C2CCN(C(C(C(CC)(C)C)O)=O)C2)C)=O)ccc(S(N)(=O)=O)cc1Cl c1(NC(C23C(CN(C(c4scc(CC)n4)=O)C2)C3)=O)cc(O)c(F)cc1F c1(CNC(c2nnnn2CC(F)F)CCOCC)ccc(C#N)nc1.C1CC1 C(N=c1ccc(S(C)(=O)=O)c[nH]1)C1C(CNC(C(C(C)C)OC)=O)C1 CCCCCC(O)C(=O)N1CCCCCC1CNC(c1cc(O)nc(SC)n1)=O CN1CCOc2ncc(C(=O)NC3(C)CC(NC(=O)C4=CCCOC4)C3)cc21 N1(C(c2cccc(OCCC)c2)=O)CCN(C(C2(F)C3CCCC23)=O)CC1CO CCC(CC(=O)N1CCC(OCCNC(C2OCC2(C)C)=O)CC1)C(C)C C1(CN(C(=O)C(C2(O)CCCC2)F)C)COCCN1C(c1cnncc1O)=O C1(C(=O)NC(C)C(=O)NC(=O)C2CC2)(NC(=O)CC2(C)CCC2)CCSC1 c1(C(N(CC(C)N(C(c2c(SCC)cccc2)=O)C)C)=O)c(C)cc(=O)oc1C C1(CCC)(NC(=O)CCC2CC2(F)F)CCCN(C(=O)C#CC(C)(C)O)C1 C(=O)(C(CCOCC)NC(=O)CCc1ccccc1)N1CCC(CCC)C1 c1(C(=O)NC2C=CCN(C(c3c(OC)nsc3)=O)C2)cnc2ccnn2c1 C1(C(=O)NC(CC(C)NC(=O)Cn2ccc(C3CC3)n2)C)CN2CCN1CC2C C1(NC(CN2C(c3ccc(CC)o3)COCC2)=O)CCCCC1(F)F C(=O)(C(C)(C)COC(C)C)N1CCC(OC(CNC(C=CC(CC)C)=O)=O)C1 CC(C)(C)CC(=O)NCCC1(NC(=O)C(O)Cc2ccc(C(F)(F)F)cc2)CC1 N1(C(C(CCn2cc(CC(COC)O)nn2)(F)F)=O)CCC12CCOCC2 CCCCCC(O)C(=O)NC1CCCCN(C(c2cscc2C(=O)OC)=O)C1 c1(C(=O)NCC(C)N(C)C(C2CCCO2)=O)cnc2ccc(Br)cc2c1 C(=O)(C(CO)C(C)(C)C)NC(C)CC1CN(C(C2COCC2(C)C)=O)C1 c1(CC)cc(C)ccc1C(N1CCCCC(CNC(=O)CC2CCOC2)C1)=O c1(C(=O)NC2CC(NC(C(c3cn(C)nc3)=O)=O)C2)cc2n(c1)CCCC2 c1(C(=O)NCC(N(C(=O)C2=CCSC2)C)C2CC2)cc2cnn(C)c2s1 c1(C(=O)NCC(CNC(C(C(CC)C)O)=O)(C)O)ccc(Cl)c(O)c1N C1(NC(C23CC(C)(C2)C3)=O)CCCN(C(c2ccc(-n3ncnn3)cc2)=O)C1 N12C3CCC1CC(C3)CC(C)C2=O.CC1CC(n2ccnn2)C1.C1(=O)C(C)N1 C1(NC(C2C(CN)CCO2)=O)CCC2CC2CC1 C12(C(=O)NCC3(F)CCN(C(c4c(CC)scn4)=O)C3)CC1COC21CCC1 N1(C(C23CCC(C(=O)OCC)C2CC3)=O)CCN(C(=O)OC)c2ccc(F)cc21 N1(C(C(Cc2ccsc2)NC=O)=O)CCC(CF)(NC(c2cscn2)=O)C1.C1CC1 N1(C(C2CN(C(c3c(C)nc(C)o3)=O)CC(C)O2)=O)CC(C)(C)OCC1C c1(C(=O)NC(CC(C)NC(c2ccsc2C(F)F)=O)C)cccn2cncc12 Cc1c(Cl)sc(Cl)c1C(N1CC(NC(C2(C)CCCCO2)=O)C(F)C1)=O c1(C(N2C(CNC(c3c(CC)n(C)cc3)=O)CC2)=O)ccc2c(c1)C(=O)NC2=O c1(C(N2CCN(C(CCCCC#C)=O)CC2CO)=O)noc2ccc(Cl)cc12 c1(OC)nc(C(=O)N(CCNC(=O)CC2(CO)CC2)C2CC2)ncc1F C1(C(=O)NCC(C)NC(C2C(c3c(C)nn(C)c3)C2)=O)Cc2ccncc2N1 c1(C(N2CCCC(C)(NC(C3C4COCC34)=O)C2)=O)cc(F)cc2c1CCC2 C1(C(C(C)C)NC(=O)C(CO)N(C)C)CCN(C(c2ccc(Cl)o2)=O)CC1 c1(CC(=O)NCC(C(=O)NC2CC2)NC(C2CC(CC)C2)=O)sc(O)nc1O CCCCC(CC)C(=O)NC(C)(C)CCCNC(C1CC12CC2)=O c1(C(N2CCN(C(=O)CO)CC2)C(=O)O)cc(F)cc(F)c1.N1CCCNC1=O C1(NC(C(CC)OC)=O)CCC(CC(=O)NC(C)CSC(F)F)CC1 C=CCCC(F)(F)C(=O)NCC1(CNC(C2CC3CC2CC3O)=O)CCC1 c1(C(N(CC(C)NC(=O)C(C)c2ccco2)C)=O)ccc2ncccc2n1 c1(NC(C(=O)NCc2cccc(SC)c2)=O)ccc(Br)c([N+](=O)[O-])c1 CCC(CC(=O)NCCC1(CNC(C2CC3C=CC2CC3)=O)CC1)C(C)C c1(C(N(CC(C)(C)CNC(C23CC(F)C2C3)=O)C)=O)cnc2ccc(F)cn12 c1(C(=O)NC2C(NC(C(C)(C)C(N)=O)=O)CCCC2)cnn2c(=O)cc[nH]c12 Cc1cn2nc(N3CC4(CCN(C(C5CCCC6C5C6(F)F)=O)C4)C3)sc2n1 C(C(=O)N1CCCC1(C)CNC(c1ccc(NC=O)cc1)=O)(C(C)C)SC c1(CC(N2C(C)CC(NC(CC(CC)(F)F)=O)C2)=O)cnn2ccccc12 C(C)(C(C)(C)C(=O)NCCC(O)CCO)NC(CN(C(=O)OCC)C)=O N1(C(CC2N(C(C(C)OCC(C)C)=O)CC2)=O)CC(C)(C)C1COC c1(OC)nc(NC2CCCCC2CNC(=O)CSC(F)(F)F)nc(C)c1F N=c1nc(CC(=O)NCc2cc(C(=O)NCCC(F)(F)Cl)cs2)[nH][nH]1 C1(SC)CN(C(c2c(Br)cnn2C(C)C)=O)CC1n1cc(C2CC(=O)C2)nn1 c1(NC(c2csc(CC3CC3)n2)=O)nc(Br)c(Br)cc1Cl c1(C(=O)NCC2(NC(c3cccc(Cl)c3Cl)=O)CCC2)ccc(Cl)c2occc12 c1cc(-n2cc(-c3cn(C4CCC(n5ccnc5)C4)nn3)nn2)ccn1 C(=O)(CCS(=O)(=O)c1ccccc1)NCC1CN(C(C(C)CC(F)F)=O)C1 C1(N(C(C=C(C)C(C)C)=O)C)CCN(C(c2cnc(S)nc2)=O)CC1 c1(C(=O)NCCC2CN(C(Cc3ccc(C)o3)=O)C2)ccc(S(N)(=O)=O)c(Cl)c1 c1(OC)ccc(CNC2COc3ccccc3O2)c2ccoc12 CC1ON=C(c2nc(C(=O)Nc3ccc(C4CCCO4)s3)cs2)C1C c1(C(=O)NCCCNC(c2c[nH]nc2-c2ccco2)=O)cccc2ccnn12 C1(C#N)(CN2CC(CNC(C3(C)CC(C#N)C3)=O)OCC2)CCOCC1 C1(C(=O)NCC2(F)CN(C(Cc3c(C)n[nH]c3)=O)C2)CC(=O)NC1(C)C Cc1cccc(Cl)c1S(=O)(=O)N1CC2CCN(c3ncc(Br)cn3)CC2C1 CCC(C)CC(C(=O)NCCc1ccc(C)cc1)NC(=O)CCc1cnc(C)o1 c1(NCCOCCC=C)[nH]c(=NCCC2(C)CCCO2)nc2c1cnn2C(C)C N1(C(c2onc(CC)n2)=O)CC2CC(NC(c3cccc(C)c3F)=O)C2C1 n1(CC)c(SC(C)CS(N)(=O)=O)nc2ccccc12.C1C(=O)N1C1CC1 c1(C(C)C(=O)N(C)CC2(O)CN(C(C3CCCC3)=O)C2)ccccc1Cl C(CC(=O)NNc1nc2cc(Cl)ccc2s1)C1CC(C)OCC1 N1(C(c2scc(-c3ccc(OC(C)C)c(F)c3)n2)=O)C2COCC1CC(F)C2 N1(C(C(COC)(F)F)=O)CC2CCCC2C1C(=O)N(CCCCC(C)C)C C(C)(CC(=O)N1CCC(OCCNC(C2SCCCS2)=O)C1)(C(F)F)N(C)C c1(C(N2CCCC(NC(C(CCO)N(C)C)=O)CC2)=O)cccc2ncn(C)c12 CC(C)C(C)(CNC(c1cnc(S)nc1)=O)NC(C1CC1C(=O)NCCO)=O N1(C(c2nccc(C(N)=O)c2)=O)CC2CC(NC(c3cccc(=O)o3)=O)C(C2)C1 C1(CNC(CC(C)C)=O)CC2CCC1N(C(=O)C=Cc1ccc(C(F)F)o1)C2 N1(C(C2(OC(C)=O)CC2)=O)CCN(C(=O)CC2CCCC(C#N)C2)C(C(C)C)C1 c1(C(N(C2CN(C(=O)C=Cc3cccnc3)C2)C)=O)cccc2cnccc12 N1(C(C=C2CCN(C)C2)=O)CCCC2(CCN(C(C3CCCOCC3)=O)CC2)C1 c1(C(=O)NCCNC(c2cc(Br)c3occc3c2)=O)cc2cccc(O)c2[nH]1 C1(N(C)C(c2cc(C(F)(F)F)cs2)=O)CN(C(=O)C2=NOCC2)CC12CC2 c1(C(=O)NCCCNC(=O)CCc2cncc(F)c2)ccc(F)c2c1OCC2 N1(Cc2ccc(C)cc2)CCC(NC(=O)CCn2c(C)csc2=O)C(C)C1 c1(C(=O)NCc2c(C(N(C3CC(CO)C3)C)=O)scc2)ccc2c(c1)CC2 c1(C(=O)NCCN(C(CC(CC)OC)=O)CC(C)O)cc(F)c(Cl)c(N)c1Cl c1(C(=O)NCC(C2CCOC2)NC(C2(C(C)C)CCCC2)=O)cc(=O)cc(Cl)[nH]1 c1(C(=O)N)cccc2c1CCO2.C(=O)(CC(=O)NC)NCCOCCN(C)C1CC1 c1(OC)cc(NC(=O)CSc2ccc(C(=O)O)c(F)c2)c(Br)nc1Br C(=O)(CCC(=O)c1ccc(Cl)cn1)NCC1(F)CC(CNC(C(C)CF)=O)C1 C1(C2(O)CCN(C)CC2)(C(=O)NC2CCCCN(C(C3(C=C)CCC3)=O)C2)CC1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NCC(CC)NC(C1CCCC(O)C1)=O C1(C(=O)NC2C=CC(CNC(CNC(N)=O)=O)C2)CCCCN1S(N)(=O)=O C1(C(=O)O)CCN(C(=O)CN2CCCCCC2)C12CC2.c1(CN)cccnc1 N1(CCC(N2CC3(CN(C(C4=C(C)CCC4)=O)C3)C2)=O)C(=O)NC(C)(C)C1=O c1(C(N(C2(c3cn(Cc4nccn4C)nn3)CC2)CC)=O)c[nH]c2nccc-2c1C CC(C)CCC(O)C(=O)N1CC2C(C(=O)NC(CCO)C3CCC3)C2C1 C1(NC(C2(OC)CCCOC2)=O)CCN(C(=O)C(=O)N=S(C)(C)=O)CC(C)(C)C1 N1(C(C2(NC(c3cc(C#N)n(C)n3)=O)C(C)CCC2)=O)CCC2CCCC12 N1(C(C(CC(C)C)O)=O)CCC(C2CCCN(C(c3ccc(F)cn3)=O)C2)C1 CCCC(CC)C(=O)N1CCN(C(c2cnc(N(C)C)cn2)=O)CC1CC1CC1 N1(C(c2ccc(C)n2C)=O)CCCN(C(C2CCCC(=O)O2)=O)C(CO)C1 CC1CN2CCCCC2CN1C(=O)C(=O)NCC(C)(C)N C(=O)(C(O)P(C)(C)=O)NCC1C(C)CN(C(c2cc(-c3ccncc3)on2)=O)C1 C1(C(=O)NCCC(CCC)O)CCCCCCN1C(=O)CSC S(=O)(=O)(c1cccnc1NCCCCN1CCCC(C)C1)CCc1cnc(C)s1 CCC(CCC(=O)N1CCC(O)C(O)C1)NC(=O)CCN1CCCC1=O c1(C(=O)NC2C(CNC(C=C(CCOC)Cl)=O)CCCC2)ccc(F)c(SC)c1 c1(C(=O)NCC(C(C)(C)C)NC(CCCCC=C)=O)ccc(N=S(C)(C)=O)cc1 Cc1nc2c([nH]1)C(C(=O)OC(c1nncn1C)C)CCC2 C=C(C)CC(C(=O)N1CC(O)CCC1C(=O)NC(C)CC(C)(C)OC)OC C=CCN=C(NCCS(=O)(=O)NCc1ccccc1Cl)NN1CCC(NC(C)=O)C1 c1(C(N2C(CNC(C(c3ccccc3Cl)OC)=O)CC2)=O)cc(C)c(F)c(C)c1 N1(C(C(C)CN2CCOCC2)=O)CCN(C(=O)CN(C)CCO)CC1 C(=O)(CC(CNC=O)C(F)(F)F)NC1CC(N(C(=O)C(CO)N(C)C)C)C1 CCCCCC(C)CC(=O)N1CCC(N(C)C(c2ccc(Br)nc2C)=O)C1 c1(CC)cc(C(=O)NCCNC(=O)C(c2cccn2C)=O)ccc1C N1(Cc2ccc(OC)c(O)c2)CCC2(CCN(C(c3cc(C)oc3C)=O)C2)CC1 c1(OC)c(C(=O)NCC(C)(C)NC(C2CC(C(C)=O)C2(C)C)=O)cnn1C c1(OC)cccc(CC(N2CCCCC2CNC(=O)Cc2cc(C)on2)=O)c1 c1(CC(=O)NC2CCC2CNC(=O)CC2(C3CC3)CC2)ccc2nc[nH]c2c1 N1(C(=O)OC)CC2CCC1CN2C(C1CCC(N2CCN(C)CC2)CC1)=O N1(C(CC(CC(C)=O)(C)C)=O)CCCC2(NC(=O)Cc3ncc(C)[nH]3)CCCC12 C(C(=O)NOCCCCF)(C1CCCO1)NC(c1cc(C(N)=O)oc1)=O N1(C(CC2(C)CCCO2)=O)CC2(NC(c3ccc(O)c(F)c3)=O)CCCC2(F)C1 N1(C(C(C)Oc2ccccn2)=O)CCOCC1C(=O)NCCc1ccc(O)nc1 c1(SC)cccc(NC(=O)CC2(C)CCN(C(c3nc(Cl)cs3)=O)C2)c1 N1(C(c2cn(C)nc2)=O)CC(NC(c2cccc3c2NCC3)=O)CC2(CCC2)C1 c1(N(C2C(C)CCCC2)C)c(F)cc(Cl)cc1N S(=O)(=O)(c1ccc(NCC2CC2C2CCC2)cc1Cl)NCCN1CCCC(C)C1 C(C)(N=c1[nH]c(=NC2CCC(C)(C)C2)[nH]c2ccsc12)c1scc(C)n1 N1(CCS(C)(=O)=O)CCOC(CNC(=O)C(c2cscn2)OC)C1 c1(C(N(CC(C)NC(=O)C(F)(F)c2nccs2)C)=O)cccc(F)c1N C1(C(=O)NCC(COC)NC(c2cc(CC)ncn2)=O)CCCC2(CCC2)C1 c1(C(=O)NCC(CC)NC(C2(CO)CCCO2)=O)c(C)cnc(OC)c1Cl CCCC(CCCNC(=O)C=Cc1ccc(CC)o1)NC(C1CCCCCC1)=O C1(NC(CSC)=O)CCCC2CN(C(c3cnn(CC(F)F)c3)=O)CC12 N1(C(c2cccc(C#C)c2F)=O)CCN(C(C2CC2(C)C)=O)C2CCCC12 C12(C(NOC(CC(C)C)C)=O)COCC1CN(C(=O)C(C)(C)CC(C)C)C2 C1(C)(NC(CNS(CCCC)(=O)=O)=O)CCC(NC(=O)Cc2ccn(C)n2)CC1 O=C1COc2c(C(=O)NC3CC4CCC3N4C(=O)CSC3CC3)cccc2N1 C1(C(N2C3C(NC(COc4cc(C)on4)=O)CC(C3)C2)=O)CN(C)CCN(C)C1 n1(CC)cc(Cl)c(C(=O)NC2CC(C)N(C(=O)Cn3cnnc3)C2)n1 C1(C(=O)NC2C(=C)C2C(C)C)(CC)CCN(C(=O)C(=O)C2CC2)C1 Cc1cc2nc(NC(=O)C(N3CC(CO)OC(C)C3)=O)sc2cc1F CN1CCC(C(N2CCOC(CCNC(=O)C3=NNC(=O)C3)C2)=O)CC1=O C(=O)(C#CC1CCOC1)Nc1cc(C(NOCC)=O)c(F)cc1 C1(NC(=O)COCCNC=O)CCC2(CC1)CC2NC(c1nccnc1C(N)=O)=O CC(C)C(CNC(=O)CN(C(=O)OC(C)(C)C)C(C)C)NC(=O)Cc1cncs1 CC1C(C(=O)NCCOCCCN(C(=O)CC=Cc2ccccc2)C)CCN1C N1(Cc2ccn(C)n2)CCC2CN(C(c3ccn4ncc(I)c4n3)=O)CC2C1 c1(-c2cn(C3C(OC)CCOC3)nn2)cc(C)c(Br)cc1C c1(OC)ccc(NC(=O)CC2CCCC(C)O2)cc1.C1(=O)C(C)CN1C(C)C N1(C(COc2cncc(C(C)=O)c2)=O)CCN(C(=O)C2=CCCCC2)C(CO)C1 C1(CNC(=O)CCC2CC2(Cl)Cl)CC2(CCN(C(=O)C(F)(F)CC3CC3)C2)CO1 Cc1c(Cl)ccnc1C(N1CCC1CNC(=O)CCCOc1cccnc1)=O c1(CC)ccc2cc(NS(=O)(=O)C3CCOCC3C)ccc2c1 c1(C(N)=O)ccc(OCC(=O)NC2CCCC(NC(C3CC(=O)N3)=O)C2)cc1 c1(C(N2CCC(NC(CCC#CC)=O)C2C)=O)noc2c1CCc1ccccc1-2 C(=O)(C(C(C)C)NC=O)NC(C(=O)N(C(CC)CC)C)c1ccoc1 Cc1ncnc(O)c1C(=O)NC(CNC(c1cnc(=N)[nH]c1)=O)C(C)(C)C c1(OC)ccc(NC(N2CCC(C)CC2c2cnn(C)c2)=O)c(Br)n1 C1(CNC(C2C(OCC)C2)=O)CCC(NC(=O)C(=Cc2ccco2)C)C1 c1(OCC(=O)NC2CCC(N(C(c3cc(C)on3)=O)C)C2)c(C)cccc1C C1(C(=O)OCC)COCCN1Cc1ccccc1-c1cccc(OC)c1 Cc1snnc1C(=O)N(C)CC1(NC(=O)CSCC(C)C)CC1 C1(C#N)(C(=O)NC2CC(NC(C(C3CC(F)(F)C3)OCC)=O)C2)CCOCC1 c1(C(=O)NCC(CNC(C2C(OC)(OC)CC2)=O)O)cc(=O)c(Br)c[nH]1 N1(C(CCN(C(CCC)C)C)=O)CC(C)CN(C(c2coc(CC)n2)=O)CC1C C(=O)(C(C)C(C)NC(=O)CCCOC(C)(C)C)N(CCCC)CCOC CCCCCC(C)NC(=O)C(CCSC)NC(=O)CN1CCC(C)C1 c1(C(N(C)CC2CN(C(CN3CC(C)C3)=O)CC23CC3)=O)cccc(S(C)=O)c1 C1(CNC(CCOCCC)=O)CCCCC1NC(=O)Cn1cccn1 c1(NC(CSCC(=O)NCCC(c2n(C)cnc2)CO)=O)ccnc2ncccc12 c1(OC)ccc(CN2C3CCCC2CC(C(=O)O)C3)c2ccccc12 CC1CCCC=C1C(=O)N1CC2CC2(C(=O)NCC(F)(F)C(N)=O)C1 N(C1CCc2cccc3cccc1c23)C1CCCC(C)C1 N1(C(COCCOC)=O)CCCC(C)(O)C1.C123CCCC1(C2)C(=O)N3 N1(C(Cc2c(C)ccs2)=O)C2CCC1CN(C(=O)Cc1cccnc1)CC2 c1(CC)ncc(C(=O)NC2CCCC2NC(=O)C(C(C)C)OC)c(O)n1 Cn1nnc2c(C(N3CC(C4CN(C(=O)C5=CCCCCC5)C4)C3)=O)ccnc12 CC1CN(Cc2nc(CC(C)(C)C)no2)CC1F N1(C(c2ccc(C#C)cc2C)=O)CCC2CCC(C1)N2C(C1(CC(F)F)CC1)=O CC(C)C(CNC(C1CC(OCc2ccccc2)C1)=O)NC(C1CC1C)=O CC(CC(=O)N(C1(C(=O)NCC2CCCCC2)CC1)C)CC(C)(C)C C(=O)(C1CCCc2c[nH]nc21)NC1CN(C(c2cc(C#C)c(C)cc2)=O)CC1C N1(C(C2C(OC(C)(C)C)C2)=O)CC(F)(Cn2cc(Cl)cn2)C1.C12(CC1)C(=O)NC2 c1(C(N2CCN(C(CNC(CC3CCC(=O)N3)=O)=O)CC2)=O)cccc(O)c1Cl c1(C(=O)NC2C(CNC(CS(N)(=O)=O)=O)CCCC2)cnc2n1CCS2 C1(NC(COCCNC(=O)OCC)=O)CCCN(C(=O)Cc2cccc(F)c2)C1 CS(=O)C1CN(C(=O)CC(O)CNC(=O)C(=O)NC2CC2)C1 Cc1c(C(=O)NC23CCC(C2)N(C(c2cccc(N)n2)=O)C3)[nH]c2ccccc12 C=C(C)CCCC(=O)NC(C1CC(NC(c2[nH]cc(C)c2C)=O)C1)C CC1(NC(c2cnc(Cl)cn2)=O)CCN(C(c2snnc2C2CC2)=O)C1 C1(O)(CCNC(COC)=O)CCCN(C(=O)CC23COC(CF)(C2)C3)C1 c1(C(=O)OC)cnn(C)c1CNC(N1CCC(CO)C1c1ccccc1)=O c1(CCNC(=O)NC(C2CCOCC2)CC)cccc(OC)c1F C(CC(F)F)(C(=O)NCc1oc(C2CC2)nc1C)NC(CC1(OCC)CCC1)=O N12CC1CC(CC)C2.c1(CC)ncc(OC)nc1CC C(=O)(C(CO)C(F)(F)F)NC1(C(N2CCC(CCC)(CO)C2)=O)CCCC1C C1(CNC(C2(CC)CC2)=O)CN(C(c2ccc(OC)nc2Cl)=O)CCC12CCC2 CC1CNC(C)CN1C(=O)C(C)(F)c1ccccc1 c1(NC(CC(C)NC(C2CCCCN2C)=O)=O)ccn2nccc2c1 C(=O)(C#CC1(C)CCCO1)N1C(CN(C(=O)OC(C)(C)C)CC)CCC1 N#Cc1cc(CN2CC(CNC(c3c(Cl)ccc(F)c3Cl)=O)C2)ccc1F C1(NC(c2cc(CC)no2)=O)COC2(CCN(C(c3nc(Br)c[nH]3)=O)C2)C1 c1(CC(C)C)c(NCCCC(=O)NCCCC(=O)OC)noc1C1CC1 c1(CC)cc(Cl)ccc1C(N1CCC(NC(=O)Cc2nnc(C)o2)C(F)C1)=O C1(NC(C(C)=C2CCC2)=O)CN(C(=O)CC23CCC(CC2)CC3)CCC1C c1(C(=O)NCC(C)(C)ONCC)ccn(C)c(=O)c1.C(=O)(C)N(CCN(C)CCO)CC O=C1Nc2c(C(N3C4CCC(C4)C3C(N3CCC(F)C3)=O)=O)cccc2C1=O C1(NC(C2C(C)CCS2)=O)CCC(NC(C2(n3nnn(C4CC4)c3=O)CC2)=O)CC1 C1(O)(C(=O)NCC(C2CC2)NC(CCCN(C(=O)OCC)C)=O)CCSCC1 N1(C(C2CCCCN2C(C2CCCC(O)C2)=O)=O)CCC(O)C12CCCC2 C1=CCCCN(N2CCN(CCC3CCOCC3)CC2)CC1 C1(c2ccccc2)(CNC(C)=O)CCN(C(=O)NCCc2ccc(C)s2)CC1 c1(OC)ccc(C(=O)N(C)CC2CN(C(c3cncc(N)c3)=O)CCO2)c(Cl)c1 C=C(C)C(C)(O)C(=O)N1CCN(C(c2cc(C3CC3)n(C)n2)=O)CC1 CC(C)CCN=C(NCCSC(C)C)NCC(c1c(F)cccc1Cl)O Cc1cc(C(=O)NCCC2CN(C(=O)CC3CCSC3)CC2C)nc(C)n1 c1(OCC)ncccc1C(=O)NC(C1CCN(C(=O)Cc2cccn2C)C1)(C)C C1(CC(=O)NCCCC(C)NC(=O)C=CCc2ccc(Cl)cc2)CCCS1(=O)=O C1(CNC(C2(COC)C=CCC2)=O)CN(C(=O)CCN2CCC2)CC1C(F)(F)F c1(-c2c(C(=O)NCCC(C)NC(c3ncccc3O)=O)c[nH]n2)ccc(Cl)cc1 c1(C(N2CCC(N(C(c3c[nH]c(=N)s3)=O)CC)C2)=O)ccc(F)cc1[N+](=O)[O-] C(=O)(C(CC)CC(C)C)NC1(C2N(C(Cc3nc(NCC)sc3)=O)CCC2)CC1 CCCC(CCC)CC(=O)NCC1CC2CCC1N2C(=O)CCC(C)(C)[N+](=O)[O-] C1(C(=O)NCCCN(C(C=C(C)C(C)C)=O)CC2CCCC2)CC(O)(C#N)C1 Cc1cccc2cc(C(=O)NC3CC4CCC(C3)N4c3nnc(C4CC4)s3)oc12 C1(NC(C2CC(OC)C2(C)C)=O)CCSC12CN(C(=O)C(F)=C(C)C1CC1)C2 C1(CN2CC(=O)OC2=O)CC2CCCCC12.c1(CC)cccs1 c1(C(=O)NC2(CNC(COC(C)C)=O)CCCC2)nc2ccc(Br)cn2n1 C1(C(N2C(c3ncc(C(=O)OC)cn3)CCC2)=O)CCC2(CCN2)CC1 N1(S(CC(=O)NC2CC2)(=O)=O)CC(OC2CCCC2)OC(C(F)(F)F)C1 c1(C(C)N(c2cc(-c3nn[nH]n3)c[nH]2)C)ccc(S(=O)(=O)F)cc1 c1(NC(CCC2(NC(CCC3C(C)=NNC3=O)=O)CCCC2)=O)ccc(Cl)nc1C c1(CC(=O)N(C2CCCC2)CCNC(CCNS(CC)(=O)=O)=O)cnc(C)s1 c1(OCCC=C)ccc(Br)c(NC(C2CC2NC(C)=O)=O)c1 n1(CCC=C)c(CC(F)F)nnc1N=c1ccn(C)[nH]1 c1(NC(C2CCOC2)CC)ccc(S(=O)(=O)N(C)CCn2cccn2)c(Br)c1 CN1CCn2ncc(C(=O)NCC3CCN(C(C4=CCSC4)=O)C3)c21 N1(C(C(C)(C)N2CCOCC2)=O)CCC2CC2(NC(=O)CC(C)(C)N(C)C)CC1 c1(C(N(CC(CC)NC(C(CC#C)O)=O)C)=O)ccn2nnnc2c1 c1(NC(c2cc(CNC(c3csc(C)c3C)=O)sc2)=O)cccc2c1OCO2 N1(C(c2c(OC)nccc2)=O)CC2(CCN(C(=O)C(C)C(=O)OC(C)(C)C)C2)C1 c1(NC(C2CC(=C)CN2Cc2ccc(C(=O)OC)cc2)=O)csc2ccccc12 CN1CCN(C(=O)CC2CC3(CC3)C2)CC1CNC(C1CCCN1S(C)(=O)=O)=O c1(C(c2n(C(CC)C)nnn2)NCc2cnn(C(C)C)c2)nn(C)cc1C c1(CCC)cc(C(N2CCC2CNC(c2cc(Cl)no2)=O)=O)c(C)o1 C(=O)(CCCCCNC(N)=O)NC1C(NC(C2CC(=C)C2)=O)C1 c1(C(=O)NCCCC(C)NC(=O)CN(C)C)ccc(CSC(F)F)nc1 C(C)(CCCCNC(c1cncs1)=O)NC(C(Br)=C(C)C)=O C1(CNC(c2ncn(C(C)C)n2)=O)CN(C(=O)CSCc2cccnc2)CCO1 C1(NC(=O)C#CC2CCOC2)CC2CC(C1)CN(C(=O)Cc1nc[nH]n1)C2 c1(OC)cccc(SCC(=O)NC2CCC(CNC(=O)CC(C)O)C2)c1 CC1CN(C(C2C(C)(C)C2(C)C)=O)CCC1NC(c1ccsc1C(F)F)=O C1(N(C(=O)CC2C=CCC2)C)CC2CCC(C1)N2C(C1COC(=O)C1)=O C1(C)(C(=O)NCCn2ncc(C(N3CC(C)(C(=O)OC)C3)=O)c2)CC(O)CN1C Cc1cncc(CCC(N2CC(n3cc(C4COCC4O)nn3)C(O)C2)=O)c1 N1(C(c2c(NC)cnnc2)=O)CC(NC(=O)Cc2cc(C)n(C)n2)CC(F)(F)C1 c1(C(=O)NC2CCN(C(CNS(CC)(=O)=O)=O)C2)c[nH]c2c(Cl)cccc12 C(=O)(C1=COCCC1)NC(C)(CNC(=O)CC1CCC(=O)O1)C1CC1 Cc1cc(=O)c(C(N2CCCC2C(C)(C)CNC(=O)CCC2CCC2)=O)cn1C CC(C)C(O)C(=O)NCC1(CC(=O)N(CCCF)C)CC1 N1(C(c2onc(C)n2)=O)CCCC(N2CCN(C(=O)C(C)(C)C3CCC3)CC2)C1 c1(C(=O)NCCN(C(=O)CCCS(C)(=O)=O)CC)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 O=C1CN(C(=O)C2=C(Cl)CC2)C(C(N2CCCC(OC3CC3)C2)=O)CN1 Cc1cccc2c(C(N3CCN(C)CC3CNC(=O)C(C)O)=O)nccc12 c1(C(N(C2CCN(C(COCC#C)=O)C2)C)=O)ccc(-c2nnc(O)n2C)cc1 C(=O)(NOCC(F)F)NCC(c1ccsc1)C c1(OC)cccc(C(=O)N(C2CCN(C(c3ccc(C4CC4)cc3)=O)C2)C)c1F C1(OC)COCCC1CC(=O)NCCN(C(=O)CCc1cn[nH]c1)CC(C)O c1(OC)cccc(C(=O)NC2CCN(C(c3cc(Cl)c(Cl)n3C)=O)C2C)c1OC C1(NC(c2c(C)c(C3CC3)on2)=O)CC2CCC(C1)N2C(=O)CCC(C)(C)C O(N1C(=O)c2cccc([N+](=O)[O-])c2C1=O)C(CCS(C)=O)C c1(OC)ccc(-n2cc(C3CN(C(c4ccccc4CO)=O)C3)nn2)c(OC)c1 c1(OC)ccc(CN2CCCC(F)(CNC(=O)CCC3CCCCC3)C2)c(OC)c1 N1(C(C(COC)N)=O)CCCN(C(=O)C(Cl)=CCl)CC1.C(C)(C)(C)OC(=O)C(=O)OCO c1(NC(=O)OC2(C(C)(C)C)CC2)ccc2c(c1)CCC2.C1CN(C)CCO1.CCO CCC(C)C(C)CONC(=O)CC1CN(C(=O)CC2CCCNC2=O)C1 C1(CC)CN(C)C(C)CO1.c12cnc(c(Cl)c1)OC(=O)NCC2.C(C(F)(F)F)O C1(C(=O)NC2CC(CO)C2)CSCCN1C(=O)C1CC1 C1(NC(C2(N(C)C)CCCSC2)=O)CC2CN(C(=O)CNC(N)=O)CC2C1 C(=O)(C(N=[N+]=[N-])C(C)C)N1CC(CCC)N(C(=O)CN2C(=O)CCC2=O)CC1 S(=O)(=O)(CCC(F)(F)F)N1CC2C(CNCc3ccc(OCC)cc3O)(C2)C1 CC1CCC(CCNC(c2cc(C3CC3)on2)=O)O1.C12(CC1)C(=O)N2 c1(C(=O)NC2(CC=C)CCN(C(=O)CCCCF)C2)cccc2nc(O)ccc12 C1(CNC(c2n(CCC)ccc2)=O)CC2CCC1N2C(c1ccc(Cl)nc1N)=O C1(C(=O)NC(COC)CO)(NC(=O)C(C)SC)CCN(C)C1 CCCC(CNC(=O)CCC(C)SC)C(=O)N(C1CC1)Cc1ccoc1 c1(CC(=O)NCCN(C(c2csc(Cl)n2)=O)CC)ccccc1OC c1(OC)ccc(C=CC(=O)NC2CCC(CNC(C3C(C)C3C)=O)CC2)cc1O C(=O)(C#CC1(C)CCCO1)N1CCN(C(c2cc(C)no2)=O)CC1CC(F)(F)F O=[N+]([O-])c1cc(Br)c(F)cc1NC(c1nnnn1CC(F)F)CCC1CCCC1 N1(C(C2(C)CCC(C)C2)=O)CCCC(C2CCN(C(=O)COC(F)(F)F)CC2)C1 C1(n2cc(-c3cccc(C(F)(F)F)c3F)nn2)(OC)CCN(C(=O)CSC)CC1 N1(C(C(CC=CCC)C)=O)CCCOC(CNC(c2cnc(OC)s2)=O)C1 C12(C(=O)NCCCOCCN(C)C(c3sccc3CC#N)=O)CC(C)(C1)C2 C1(C(C)NC2CC(C(C)(C)C)C2)CCCCCC1 c1(C(=O)NCC(c2ccccc2F)NC(C(C)(F)F)=O)ccccc1N=[N+]=[N-] C(CCC)(C(=O)N1CCCC1C=CC(N1CCC(OCCF)C1)=O)=CCC C(C)(CC(=O)NC1CCN(C(=O)CCc2ccoc2)CC1)(C(F)(F)F)N(C)C N1(C(c2ccc(SC(C)C)cc2)=O)CCC(NC(=O)Cc2ccsc2)C(C)C1 c1(C(=O)NC(CN(C(c2ccnc(C)c2)=O)CC)C)ccc(F)c(C)c1N C1(CC=C)(C(=O)NC2CCCC2CC(=O)NC2(CCOC)CCC2)CCOC1 c1(C(=O)NC2C(C=C)CN(C(C3CC3C(C)(C)C)=O)C2)ccc2c(c1)CCO2 C1(C(N(CCCN(C(CCN(CCOC)C)=O)C)C)=O)CCCC(OC)C1 C(CC(CO)C(C)C)NC(c1c(C)nc(CNC(c2ccc(O)nn2)=O)o1)=O c1(OC)cc(OC)c(C(=O)NCC23CC(NC(=O)CSCC)(CCO2)C3)cc1N.OC C1(C(CC)(O)C)CCNCC1.C(=O)(CNC(=N)O)N(C)CC CC1CN(C(c2cccc3nncn23)=O)C(C)CN1C(c1cnc2n1CCS2)=O N1(C(C2N(C(C(CC3CC3)OC)=O)CCC(C)(C)C2)=O)CCC2(CNC(=O)C2)C1 N1(C(c2cccc(C(F)(F)F)c2)C)CCC(C(C2CCCO2)O)CC1 c1(C(N(C(C)C(=O)N(C2CC(CO)C2)C)CC)=O)cc(C)cc(C#N)c1 C=CC(F)(F)C(=O)NC1CCN(C(=O)NC2CC(OCc3ccccc3Cl)C2)C1 CN1CCCC1CC(=O)NCC(C)(O)CNC(=O)CCc1cnc(C2CC2)o1 Cc1c(Br)ccc(C(=O)N(CC(O)CN(C)C(c2ccc(Cl)[nH]2)=O)C)c1N C1(NC(CC2(NC(C)=O)CC2)=O)CN(C(=O)C2=CCSC2)CCC1C CC1CN(C(c2c(Cl)c(C(F)(F)F)nn2C)=O)CC(C)(C)C1 N1(C(C(=O)NC(C)C)C2CC2Cl)CCCCC1CC1CCC1 C1(C)(C(=O)NCC(C)(C2CC2)NC(=O)C(=O)NCC2CC2)CCCNC1=O N1(C(c2cc(C)cc(O)c2)=O)CCC(C2CC2)C1C(=O)NCCCSC(F)F O=C(C1=COc2ccccc2OC1)NCC1CC1NC(c1ccn(C2CC2)n1)=O C(=O)(C1CC(=O)Nc2cc(F)ccc21)OC(C(C(C)C)CC1CCCC1)=O C1CN(C(c2ccnc(NC3CCOC3)c2)=O)CCC1C(F)(F)F c1(C(=O)NCCCNC(CCC)=O)cnc(C)c(Cc2ccc(F)cc2)c1 c1(N(CC(=O)NCC(CC)NC(=O)C2=CCCC2)C)ccc(Cl)cc1 N1(C(c2nc(NC(C)=O)sc2)=O)CCCC(C)(C(=O)Nc2nncs2)C1 C(C)(CO)(C(=O)N(CCC(=O)N(C)CC1CCN(C)CC1)C)OC c1(NCC2(OC)CCSCC2)ncc(C)cc1S(=O)(=O)NCC1CC(=C2CC2)C1 Cn1ccnc1S(=O)(=O)N1CCN(C(=O)C(C)(C)NC(=O)OC(C)(C)C)CC1 C1(NC(c2n(C(CC)C)nnn2)(C)COC2(C)CCSC2)CC2(CCCCC2)C1 C1(NC(C2(CC=C)CCC2)=O)CC(NC(c2cccnc2N)=O)C(O)C1 C1(NC(CCOCCOC)=O)C2CC1CN(C(C1CCC(O)CC1)=O)C2 C1(CCC#C)CCCN(C(=O)CCN(C)C(c2cc(CC)ccn2)=O)C1 C(c1ccc(F)c(F)c1)=CC(=O)NCC12C(CN(C(c3nnc(C)s3)=O)C1)C2 c1(C(=O)NCC(CC)NC(C(CC)SC)=O)sc(CC(F)(F)F)nc1C N1(C(CC2N(C(C(n3ccc(C)n3)C)=O)CC3(CC3)C2)=O)CCn2nncc2C1 C1(CC)CN(C(c2cn(C(F)F)cn2)=O)CC1NC(c1cc(OC)n[nH]1)=O C1(C(C)OC)CCN(C(=O)CCC(C)NC(c2cc(OC)n[nH]2)=O)CC1 C(=O)(C#CC(C)(C)C)NC(CCOCC)C(=O)N(C)Cc1c[nH]nc1C C1(CNC(C(C=CCCC)O)=O)CC2(CC2)CN1C(=O)C.c1(C)nc[nH]n1 C(=O)(C(CCC1CC1)NC(=O)N)OC(c1csc(-c2ccsc2)n1)C.C(C)(C)(C)N C12(NC(C3CC(CCC)C3)=O)CCCC1N(C(=O)C(C)C)CC2 c1(OC)cc(C)c(C(N2CCCCC(NC(=O)C3=C(C)OCC3)C2)=O)c(F)c1 C1(NC(C(CCOC)C)=O)CCC2(CC1)CN(C(c1cccc(C#N)c1F)=O)C2 c1(CNC(CS(CC)=O)=O)cc2n(n1)CCN(C(c1coc(COCC)n1)=O)C2 C1(O)(CCNC(C=C2CCN(C)C2)=O)CCN(C(C2(C)CC=CC2)=O)C1 Cc1c(C(N2CCC(O)(C(C)CNC(=O)COCC3CCCC3)C2)=O)nnn1C c1(C(=O)NC(CC(C)C)CNC(=O)C=Cc2ccc(C(F)F)o2)nnc(O)cc1O Cc1cnc(Cl)c(NC(C2CCN(C(=O)CCc3cnccn3)CC2)=O)c1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C(C2NC(=O)C(F)C2)=O)CCC1 c1(C(C)(C)C)n[nH]c(=NCC2CC(NC(c3cnc(Cl)[nH]3)=O)C2)o1 C(N=c1nc(SC)[nH]c(=NC2CC(C)(C)OC(C)(C)C2)[nH]1)C1(C)N=C(C)SC1 c1(CC)cc(Br)ccc1C(=O)NCCC(C)CCNC(=O)CSC C(=O)(C(CO)c1ccccc1)N1CC(CCNC(=O)CNC(C2CCCC2)=O)C1 N1(C(C2=C(C)OCC2)=O)CC(C)CN(C(c2cscc2C)=O)C(C)C1 c1(C(=O)NCC(C)NC(=O)C2=NOC(C)(C)C2)cc(Br)c(F)cc1Cl c1(-c2cc(C(=O)NCC3(OCC)CCCOC3)n[nH]2)cc(F)c(C(F)(F)F)c(F)c1 c1(CC)cc(C(=O)NC2CN(C(=O)C(=C3CCCCC3)F)C3CC23)ccc1Cl c1(C(=O)NC2CC(NC(c3cn(CC)nn3)=O)C2)ccccc1NC(C)C Cc1ccc(O)cc1C(=O)NC1CN(C(=O)CCCN(C)C)CCC1C(F)(F)F c1(C(=O)NC(C2CN(C(C3CCC4CC34)=O)CCO2)C)ccc(CC(C)C)nc1 CCC(C)(C(=O)NCC#CCNC(c1ccc(C(=O)OCC(F)(F)F)nc1)=O)OC C(=O)(CC(C)(O)CNC(=O)C1=CCN(C)C1)N1C(CCC)(CO)CCC1 c1(C(=O)NC2C(C)N(C(=O)CNC=O)CCC2)ccc(P(C)(C)=O)cc1 C12(C(=O)NC(C)CCNC(c3ccc(CCF)cc3)=O)CCC(C1)S(=O)(=O)CC2 C1(CNC(Cc2c(C)occ2)=O)CCC(C(=O)NCCC2NC(=O)NC2=O)CC1 N1(C(c2c(C)nco2)=O)CC(C)(C)OCC1CNC(c1c[nH]c2ccncc12)=O C12(NC(=O)Cc3cc(F)cc(F)c3)CCN(C(=O)C=Cc3ccco3)CC1C2 c1(OC)ccnc(CNC(=O)C(C(C)C)NC(c2ccoc2Cl)=O)c1 c1(C(=O)NC2CCCC(NC(C(C)N(C)C)=O)CC2)ccc2c(c1)N(C)C(=O)C2 C(CC1CCCC1)(CC(=O)N(CC(C)C#N)C)NC(C(C)SCCCC)=O CC1(C)C2CCC1(C)C2C(=O)NC1C2CN(C(c3cc(Br)cnc3O)=O)CC12 C1(c2cn(CC(=O)N)nn2)CCCS(=O)(=O)C1.C1(C(=O)OC)CCC(F)(C(=O)O)C1 N1(C(c2ncn(C(C)C)n2)=O)CCOC(C)(C(C)C)C1.C12(CC1)CC(=O)N2 c1(C(=O)NCC2(CCNC(C3COCCO3)=O)CC2)cc(F)c2[nH]nnc2c1 C1(CNC(c2c(C)occ2)=O)CC(C)(C)CCC1NC(=O)CSCc1cscn1 CCCCC(CNC(c1cncnc1CC)=O)NC(=O)CC(C)SC C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCOC1CN(C(c2cc(O)cs2)=O)C1 C(=O)(C(C)(C)C(C)(C)O)N1CCN(Cc2ccc(OC)cc2)CC1 C(C)(C(C)(C)C(=O)NCCC(O)CCC)NC(C(CC=C)C)=O C(=O)(C1=NNC(=O)CC1)NCC(CCNC(Cn1nc(C)oc1=O)=O)O C1(CNC(c2cn(CCC)nc2)=O)CC(C)CCN1C(c1nnccc1C)=O N1(C(C2N(CC)CCCC2)=O)CCC(NC(C)=O)C(C)(C)C1 CC1(C(=O)NCCC2C=CCC2)C=CCN1C(c1ccncc1)=O Cn1cc2ncc(C(=O)OCC34CCCC(C)(C3)OC4)cc2n1 c1(CCC(=O)Nc2c(C)cc(C(CSCCC)=O)o2)ccc(C(=O)OC)c(O)c1 Cc1cc(CN2CCCCC2c2nnc(-c3cccnc3)o2)ccc1Br N1(C(Cc2cn(CC)nc2)=O)CCC(CNC(=O)COCCOC)C(C)C1 Cc1cc(C(=O)NCCCCCn2cc(CCN(S(C)(=O)=O)C(C)C)nn2)cs1 c1(C(N2CC(OCCCNC(C3(CO)CCC3)=O)C2)=O)ccc2c(c1)CCCC2 C1(CC#C)(C(=O)NC2CCCCC2CNC(c2snc(C)c2N)=O)CC=CCC1 N1(C(=O)NCC2CCC(C)(CC)O2)CCc2nn(C)c(N)c2C1 c1(NC2CCCC(C#C)C2)nnc2cccnc2c1N C1(CC(N2CCC(COC)(NC(=O)Cc3cncs3)C2)=O)CCCC(C)(C)C1 c1(C(C)=O)ccc(OCC(=O)NC(C)C(C)NC(c2cnn(C)n2)=O)cc1 c1(C(=O)NC2CN(C(C3CCC(=O)C3)=O)CC2O)ccc2sc(O)nc2c1 C1(C(=O)NCC(=C)CCNC(c2coc(C(F)F)c2)=O)CC2CCC(C1)S2(=O)=O N1(C=O)CCC(O)(C(F)(F)F)CC1.c1(CC)ccccc1OCC(=O)NCC(C)(C)C C1(C(N(C2CCN(CC)C2)C)=O)CC2CCCC2N1C(c1[nH]cc(C)c1C)=O CCC(C)(CO)C(=O)N1CCC(C(C(C)C)NC(c2cnc(O)o2)=O)CC1 CC12CCC(C(=O)NC3CN(C(=O)CCc4ccc(C#N)cc4)C3)(C1)OC2 C1(NC(COc2cc(CC)on2)=O)CN(C(C2(C(F)F)CCCO2)=O)CC1OC c1(C(=O)NCCCCCNC(C2CCS(=O)(=O)N2)=O)ccc(-n2cccn2)nc1 N1(C(C=CCN)=O)Cc2ccccc2C1CNC(=O)CN(C1CCC1)C.CC=CCl c1(SC)nn(C)cc1C(=O)NC1CC(N(C(=O)CC2(C(F)(F)F)CC2)C)C1 c1(C(N(CC#CC(F)(F)F)C)=O)ccnc(Cl)c1F n1(CC#C)cccc(NC(C2(CC)CN(C(=O)C(C)CC(C)C)C2)=O)c1=O C12(NC(COC(CC)C)=O)CCC(CC1C(=O)NCCOCCSC)C2 Cc1cccc(OC(C)(C)CNC(=O)NNC(c2cccc(=O)n2O)=O)c1C C1(NC(CSCC#C)=O)CCCN(C(=O)CC2CCC(=O)N2)CCC1 c1(C(N2CCC(CN(C(=O)CC3=CCCC3)C)C2)=O)cncc(C#N)c1 C12(C(=O)NCCCCC#C)CCCC1N(C(=O)Cc1nnc(S)n1C)CC2 C1(C(=O)NCCC(C(C)C)OC)CC2CN(C(C34CCC(C3)OC4)=O)CC2C1 N1(C(C2(C)CCC(C)C2)=O)CC2CCCN(C(c3cnc(O)o3)=O)C2C1 Cc1cnc(C(=O)NC23CCN(C(c4cc(Cl)ccn4)=O)CC2C3)cc1C c1(OC)ncc(C(=O)Nc2ccc(F)cc2)c(OC)n1.C1(=O)CC=CCN1 N1(C(CSc2c(C)noc2C)=O)C2CCC1CC(CNC(=O)CC=C(Cl)Cl)C2 c1(C(Cc2ccccn2)NC(c2c(C)csc2C)=O)cccc2ccccc12 C(CCN=C(NCc1cc2ccccc2s1)NCC(c1ccoc1)O)OC(C)C C(C(C(=O)NCc1nc(CO)n[nH]1)NC(c1cc(C2CC2)no1)=O)N(C)C c1(C(=O)NC(CC)CNC(C2(C)C=CCCC2)=O)cccc2oc(=N)[nH]c12 c1(C(=O)NCC(CNC(c2cnc(S)[nH]2)=O)OC)coc(C(C)(C)C)n1 c1(CC(N2CCC(O)(C(C)NC(CSC(C)C)=O)C2)=O)cc2ccccc2o1 c1(N(C)CC2CCOC2)nc(=NCC23CCCC2C3)[nH]c2cccc(F)c12 N1(C(COCCOCC#C)=O)CCC(F)(CNC(C2CC23CCCC3)=O)C1 N#CC1CN(CC(=O)NCCc2ccns2)CC1c1ccccc1 C1(CCNC(C(C)SC)=O)CCCN(C(=O)CCOc2ccc(F)cc2)C1 Cc1cc(Cl)c(C(N2CCCC(C(C)NC(=O)C(c3ccncc3)C)C2)=O)cn1 Cc1csc(C(=O)NC(C2(C(N3CC(C#N)C3)=O)CC2)C)c1C C1(C(N2CCN(C(=O)CSCC(F)F)C(C3CCCC3)C2)=O)CCS(=O)(=O)CC1 C1(C(=O)NCCCCCCOC)CN(C(=O)CCCC(C)C)CC(C)(C)C1 N1(C(C(C2CCN(C(=O)COc3ccsc3)CC2)C)=O)CCCC12CCC2 CC(C)C(C)C(C)CC(=O)N1CC2CCCC(C1)N2C(C1(O)CCSC1)=O CCCC(C)CC(=O)N1CCN(C(=O)CC2CC=CC2)CC1COC c1(C(=O)NCCCNC(C2CCCC(C)C2)=O)nccc(Cl)c1Cl C1(C)(CNC(C(N2C(=O)CCC2=O)CC)=O)CCCN(C(=O)CC(=O)N(C)C)C1 c1(C(=O)Nc2c(C(=O)OC)scc2)cccn2c(-c3cccc(O)n3)cnc12 C1(c2n(C(C(=O)OC)C)nnn2)(NCc2cncn2C)CCSCC1 c1(C(N(CC(C)(C)CNC(=O)C(n2ccc(C)n2)C)CC)=O)snc(C)c1N CCC(CC(=O)N1CC(CN2CCN(C(c3sc(C)nc3C)=O)CC2)C1)C(F)F c1(C(=O)OC(C)C(=O)Nc2cccc(Cl)c2)cc2nnn(C)c2s1 C(C(CC(C)C)NC(c1c[nH]nc1C(C)(F)F)=O)NC(c1ccc(SC)s1)=O C1(n2cc(COC)nn2)CCN(C(c2cn(-c3ccccc3F)nn2)=O)CC1 c1(OCC)ccccc1C(=O)C(=O)N1CCC1CNC(C1CCCCO1)=O C#Cc1ccc(C(=O)NC(C)(CO)C(=O)N(C)Cc2noc(C)n2)c(C)c1 Cc1ccc2c(c1)CCC(C(=O)NCC#CCNC(c1ccc(F)cc1C)=O)O2 C1(CNC(C2C(C)C2)=O)CCC2CN(C(c3cc(C#N)on3)=O)CCC2C1 N1(C(Cc2cc(CC)no2)=O)CCC2CN(C(=O)CN3C(=O)CCC3=O)CC2C1 C(N=c1[nH]c(NCC(C(C)C)C(C)C)nc(=N)[nH]1)c1cccc(CNC(C)=O)c1 N1(CC(=O)N(CC(=O)NCCC2COCCO2)C2CC2)CC2CC2C1 Cc1csc(NC(C)C(=O)N2CCC2CNC(=O)CC2COC(=O)C2)n1 c1(CC(=O)NCCC2CCCSC2)c[nH]c2cc(O)ccc12 C12(CC)CN(C(c3ccncc3)=O)C(CNC(=O)CN(C3CCSC3)C)(C1)C2 c1(C(=O)NCC(c2ccccc2)NC(CNC(CC)=O)=O)cncc(C(N)=O)c1 C(=O)(C(C)P(C)(C)=O)NCC1CC(F)(CNC(C(C)OCC=C)=O)C1 C1(C(=O)NCC(CCNC(=O)CN(C)S(N)(=O)=O)OC)CCCCC(=O)N1 N1(C(c2ccc(=NCC)[nH]c2)=O)CCCC12CCN(C(C1CC1Cl)=O)CC2 C(CC)(C(=O)N1CCC(CCC(=O)NC2(C(F)F)CCC2)C1)OCC Cc1nnc2ccc(C(N3CCC(CNC(C4C(C)C4C)=O)C34CC4)=O)cn12 C1(C(=O)NCCOC2CCN(C(C3CCC(O)CC3)=O)C2)CCn2cncc2C1 c1(OC)cc(OC)c(C(N2CCCC(CNC(=O)COC(C)=O)C2)=O)cc1Br C12CCCC(O1)C(=O)OC2.N1(C(=O)OC(C)(C)C)CCC(=CC(=O)OC)C1 c1(C(N2CCC(CN(C)C(c3cc(C4(C)CC4)on3)=O)C2)=O)cc(C#N)cs1 C1(CNC(c2ccc(CC)[nH]2)=O)CN(C(=O)C(C)(C)CSC)CCCO1 N1(Cc2n(CCC)nnn2)CCOC(C)(CNC(c2sc(COC)nc2C)=O)C1 c1(CC)ccccc1C(=O)NCc1cc(CNC(=O)CSC(F)(F)F)no1 N1(CC)CCC(NC(c2sccc2CNC(=O)COC2(C)CCC2)=O)C1 N1(C(C(C)O)=O)CC(CCNC(c2cnn(Cc3ccccc3)c2Cl)=O)C(C)C1 c1(C(=O)NC2C(CNC(c3cn(C)c(=O)n3C)=O)C2)nccn2ccnc12 c1(C(N2CC3CN(C(C4CCC(C)O4)=O)CC3C2)=O)ccnc2c1ncn2C CCC(CC1CCC1)C(=O)NCC1(NC(=O)CN2CCCCC2C)CCC1 C1(CC)CN(C(=O)C(C)SC(F)(F)F)CCN1C(c1cnc(C)o1)=O C(=O)(CCCC(CC)CC)N1CC(C(N2CC(CC#C)OCC2)=O)C1 c1(C(=O)N(c2ccc3c(c2)OCO3)Cc2cscc2Br)cc(Br)c2ccccc2n1 N1(C(c2c(CC)c[nH]c2)=O)CC2CCN(C(c3ocnc3C(F)(F)F)=O)CC12 N1(CC(CNC(C(C)N(C)C)=O)O)CC(NC(=O)C#CC2CC2)C(C)(C)C1 c1(OCC(=O)NCCc2cn(-c3nccc(OC)c3)nn2)ccc(Cl)cc1Cl c1(C(=O)NC2C(CNC(C(F)(F)C3(OC)CCC3)=O)CC2)cncc(C)c1 c1(OC)cc(C(N2CC3CC2C3C(=O)NCc2ccccc2O)=O)nn1C CCCC(C)(CC)C(=O)NCC1CN(C(=O)C=C(C)c2ccco2)CCC1C c1(C(=O)NCC2(O)CCN(C(CSCC)=O)CC2)nccc2cc[nH]c12 N1(C(C=CCOC)=O)CC2CCCC(Nc3nc(Cl)nc(C)c3Cl)C2C1 N1CC(n2cc(CCCCCO)nn2)C2CCCCC12.CS(=O)(=O)CCCO C1(C2CCC2)(C(=O)NC(C2(O)CCN(c3cc(=O)n(C)cn3)C2)C)CC1(F)F CC1(C)CN(C(C2CC2C(F)F)=O)CC1CO.c12ccc(c(F)c1)CN(CC)C2=O C(=O)(C(CCC)CC(C)C)NC(CC=C)CC(=O)NC(CC(=O)OC)C1CC1 C#CCCCC(C)C(=O)N1CCOC(CN(C)C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 c1(COC)ccc(C(N2CC(CO)(NC(c3csc(-c4cnc[nH]4)n3)=O)C2)=O)o1 N1(C(C=C(CCC)C)=O)C2CC=C(C(=O)NC(C)C(C3CC3)OC)C1CC2 N1(C(=O)CCC2CC2)CCC2C(CCCN2C(=O)C(C2CCS(=O)(=O)CC2)O)C1 C1(NC(CC#N)=O)CCCC(CNC(C2(CC3CC3)CCCO2)=O)C1 Cc1nc(C(C)C)nc(N2CCC(CNC(=O)CCN3CCC(F)C3)CC2)c1Br C1(C(=O)NCC(=O)NCC=C)CCC=CC1NC(C12CC(C#N)(C1)C2)=O Cc1cc(C(=O)NC2CC(C(C)NC(=O)C(N3CCCCC3)C)C2)no1 C(C(=O)NCCSC1CC1)(C(C)C)OC(C(=O)N)C.c1(OCC)ccc(COC)cc1 C1(CNC(c2ncn(CC)c2)=O)CCCCC1NC(C1(SC)CCC1)=O c1(C(N2C(CNC(C3(C(F)F)CC3)=O)CC(OC)C2)=O)nccc(Cl)c1C c1(CNC(C(CCOCCC)OC)=O)cccc(CC)c1.C12(CC1)CC(=O)N2 c1(CN(C)C)ccccc1C(=O)NCC(O)CNC(c1cc(Cl)cn1C)=O CCC1N=C2N=c3ncn(C)c3=C(N2)N1.C1(NC(=O)C2CC2)CCN(CC2CC2)C1 c1(OC)ccc(NC(C2CC2NCc2ccc(C(N)=O)cc2)=O)cc1N(C)C C1(C)(C(=O)NCC(N(C)C(c2cccc(C3(O)COC3)c2)=O)C2CC2)CC2(CC2)C1 N1(C(c2n(C)ncc2)=O)CCCC2(CCC(NC(=O)CCCN3CCCC3)C2)C1 Nc1ncc(Br)cc1C(=O)NCC(C(=O)O)c1cn[nH]c1 Cc1cc2occc2c(=NC(CCO)C(F)F)[nH]1 CCCCCCCCC(=O)NCCC(C)N(C(=O)C1=CC2CCCCCCC12)C c1(CCC(N2C(CNC(C(CCSC)O)=O)CCCC2)=O)ccccc1[N+](=O)[O-] C1(NC(CCSCC)=O)CC2CC1CN(C(=O)CCN1CCCCC1=O)C2 C1(CC(N2CC(OCC(=O)NC3CCCCS3)C2)=O)CC2C=CC1C2 c1(CC)sc(=N)[nH]c1C(N1CC(=C(F)CNC(=O)CSc2ccccc2)C1)=O N1(C(=O)NC(c2nc3ccccc3[nH]2)CCC)CCC(C#N)(C#N)CC1 C1(C)(COC)CC(NC(c2cnc(OC)c(Cl)c2)=O)CN1C(=O)C(C)=C1CC1 N1(C(C(C)C2CCCO2)=O)CC2CCCC(C1)N2Cc1ccccc1 C1(C)(CNC(c2c(C)nco2)=O)CN(C(C2(C3CCCCO3)CCC2)=O)CCO1 C(=O)(CC(C)CC(=O)NCC1CCCC1NC(c1cnc2scnc2c1)=O)OC c1(CC(N2C(CN(C)C(C3CC(C)N(C)C3)=O)CCC2)=O)ccc2c(c1)CCC2 c1(C(N)=O)nc(C(=O)NC2CC(CNC(c3cc(C(F)(F)F)ns3)=O)C2)cs1 c1(OC)ncc(CN2CC(NC(=O)CCN3CCN(C)CC3)C(F)C2)cn1 N1(C(CN=[N+]=[N-])=O)CCCCC1CC(=O)N(CCC(F)(F)F)CCO CCC(CC(=O)NC1CCCC1C(=O)NCC1(OC)CCC(C)C1)C(C)C Cc1nc(-c2ccccn2)nc(C)c1C(=O)N(c1nnccc1C#N)C(C)C C1(N(C(c2ccc(CSC)o2)=O)C)CCCN(C(=O)C(F)(F)c2cncs2)C1 CCCC(O)C(=O)NC(CCC1CC1)C(=O)N(C)Cc1ccc(C2CC2)o1 C(C)(C)(CCCC(=O)N1CCC2(CC1)CC2)NC(C(CCC)SC)=O N1(C(c2c(C)n(C3CC3)nc2)=O)CCC2CCC(C1)N2C(C1CC12CC(O)C2)=O C(CC1=CCOCC1)NC(c1cccc(F)c1C(N)=O)c1n(CCCC)nnn1 C1(C(N2CC(CCC)C(NC(=O)CC3CCCC3)C2)=O)CCOCC12CCCC2 C1(C(=O)NC(CC(C)C)CNC(=O)CC2(O)CCCC2)CS(=O)(=O)CC(=O)N1 N1(C2CN(C(C(C)CO)=O)C2)CCN(C(=O)CC2(O)CCOC2)CC1 Cc1cccc(C(F)(F)C(=O)N(C(C)CNC(C2(n3cc(Cl)cn3)CC2)=O)C)c1 N(C(=NCC1CC(n2cncn2)C1)N(C)Cc1ccco1)C(C)Oc1ccccc1 C1(CNC(C(CC)NC(N)=O)=O)CCC2(CCN(C(C3(C(N)=O)CC3)=O)CC2)O1 N1(CCSC)CC(C(=O)NC(CNC(c2cc(=O)cc[nH]2)=O)C(C)(C)C)CC1=O C(CCN(C(=O)C1=CCSC1)C)(C(C)C)NC(C(CC)C1CCCCC1)=O c1(C(N2CC3C(CNC(C4C(C#C)C4)=O)C3C2)=O)ccc(C)c([N+](=O)[O-])c1 c1(CCC(=O)NC2CCC23CN(C(C2CCO2)=O)C3)c[nH]c2ccc(F)cc12 N1(C(C(C2CC(NC(c3nn(CC)nc3C)=O)C2)F)=O)CC(=O)NC(=O)C1 C(C(C(=O)Nc1c(O)cccc1F)C(C)(C)C)NC(COCC=C)=O C1(N(C(C(CC)(F)F)=O)C)CCCN(C(=O)C(C2CCCC2)OC)CC1 N1(C(CC(C(=O)OC)(C)C)=O)CC(C)CN(C(=O)CC2CCCCC2O)CC1C CCCCCC(O)C(=O)NCCOCCC(=O)N(CC(C)OC)C N1(NC(C2OCCC(=O)C2)=O)CCCC2CCCCC12.C12(C(=O)O)CC(CO1)C2 CC(C)CC(O)C(=O)NCCC(C)NC(c1ccc(C#N)s1)=O C1(C(N2CCCC(CCNC(C3CC(SC)C3)=O)C2)=O)CCC2(CCC2)CC1 C#CCC(C(=O)NCCc1cscn1)NC(C1CC(C)=NO1)=O CN1CCC(n2cc(C(=O)NC3COCC3CNC(=O)CCCF)cn2)CC1 c1(C(N2CC(NC(C(C)OCCC=C)=O)C(OC)C2)=O)cc(C)c(Cl)cc1C C1(C(=O)NC(C)CN(C)C(c2cccc(CN=[N+]=[N-])c2)=O)CCC(C)(C)OC1 N(C(=NCc1ccc(OC)cc1)NCC1COC(=O)O1)CC(C)(CO)NC N1(C(C)CO)CCCN(C(=O)NCc2ccc(Sc3ccc(Cl)cc3)cc2)CC1 C1(NC(c2cc(OC)nc(Cl)c2)=O)CN(C(c2ccc(Cl)cn2)=O)CC2(CC2)C1 N1(C(c2cc(CC)c(C)cc2)=O)CC2(CCCC2NC(=O)CCCCCOC)C1 C1(COC)(CNC(c2ocnc2C)=O)CCN(C(C2CC3(CCC3)C2)=O)C1 c1(-c2nc(CCCC)nn2CCOC)cc(N)ccc1C N1(C(COCC)=O)CCC2(CC1)CN(C(=O)CCOC(=O)CNS(=O)(=O)NC)C2 N1(C(C)C)CCCC(N=c2[nH]c(=NCC(C)(C)N(C)C)[nH]c3c2CSC3)C1 CCCCS(=O)(=O)NC(C)C(=O)NCCC(C)NC(c1cnc(C(F)(F)F)s1)=O Cc1cnsc1C(=O)NC(C)CC1CN(C(=O)C=CCn2cncn2)C1 N1(C(Cc2cccc(C#C)c2)=O)C2CCC1CN(C(=O)CC1CC=CCN1C)C2 c1(C(=O)NN(CC)CC)ccc(-c2ccc(N(C)C(C3CCC3)C)nn2)cc1 N1(C(CNC(CC)=O)=O)CCC2CC12C(N1CC(N2CC(F)C2)C1)=O N1(C(c2c(CCCC)onc2)=O)CCCCC(CNC(=O)C=CCF)C1 CC(C)(CC(=O)NC1CCC1NC(=O)CCCOC(C)(C)C)c1ccccc1 C=CCC(F)(F)C(=O)NC1CCN(C(c2ncc(C(F)F)s2)=O)C(C)C1 CCC(C)(CO)C(=O)NC1(CNC(=O)CC2(CC(=O)OC)CCCC2)CCC1 CCCC(C)(CC)C(=O)NC1CCCN(C(=O)COc2cccc(Cl)c2Cl)C1C c1(C(=O)NCCC2N(C(C(=Cc3cccs3)C)=O)CCC2)cccc(C2CC2)c1 C1(C(=O)NCc2cn(CC3C4CCCC34)nn2)CCCCCCC1 Cc1nc(C(N2CCC(c3cc(CNC(C4CN(C)C4)=O)on3)CC2)=O)c(C)o1 c1(CC)cncc(C(=O)NCC(C)(O)CNC(c2cc(C3CCC3)no2)=O)c1 N1(C(CC(C)OC)=O)CC2(C1)CN(C(=O)Cc1ncn(C)c1C)CC2CO C1(C(N(CC#C)CC)=O)CC2CC1CN(C(=O)C1=CCC(C)CC1)C2 C(=O)(C(C)(C1CC1)N(C(=O)C(C)OCC=C)C)NC(CC#C)C C(C)(C12CC3CC(CC(C3)C1)C2)=CC(=O)NCC(CNC(C(CC)F)=O)(C)O C1(C(=O)Nc2cccc(C)c2)CC2CN(C(=O)CCC3CCCOC3)CC2C1 O=C(CC1CCc2ccc(O)cc21)Nc1cc(Br)c2cn[nH]c2c1 N1(C(C=CCOCCOC)=O)CCCN(C(c2c[nH]c(=N)o2)=O)CC1C C1(CNC(c2c(C)nc[nH]2)=O)COCCN1C(=O)Cn1c(C)csc1=O C1(CNC(Cc2c(OC)c(F)ccc2)=O)CC2(CCN(C(C)=O)C2)CO1 C1(CCC)CN(C(=O)C=CCCC(C)C)CCN1C(=O)C(C)(C)COC Cc1ccc2c(c1)CCN2C(c1cc(CCNC(=O)C(C)C2CC2)on1)=O N1(C(C(C(CC)O)(C)C)=O)CC2CC(C)N(C(=O)CCC3CCCN3C)C2C1 C(=O)(C1CCc2cccc(=O)n21)NC1C(NC(c2ccc(OC)cc2C)=O)C1 C1(NC(=O)NC)CCC(N=c2ccnc(C(C)(C)C)[nH]2)CC1 c1(C(N2CC(CNC(C3(C)CC3(F)F)=O)C2)=O)cccc2c1COCC2 C1(S(C)(=O)=O)(C(N2CCC(C(C)NC(=O)CC3CN(C)C3)CC2)=O)CCCCC1 C1(NC(=O)CCCC2CCC2)CC12CCN(C(C1CCN3CCCC3C1)=O)CC2 C1(C(=O)NCCC)CN(C(=O)C#CC2CCC2)c2ccccc2O1 CC1COc2ccc(C(=O)N(C3CN(C(=O)C(C)CC(C)(C)C)C3)C)cc21 c1(C(=O)NCCCN(C)C(C2(N(C)C)CCCC2)=O)cc2n(n1)CCCO2 Cc1cc(=NCCC2CCS(=O)(=O)C2)[nH]c(C(F)(CF)CF)n1 c1(OC(C(C)NC(=O)C(C)(C)Oc2ccccc2OC)=O)cccc(C#N)c1 c1(C(=O)NCC(C)(CC(C)C)NC(c2c(C)nco2)=O)cc(S(N)(=O)=O)co1 Cc1nc(CO)ncc1C(=O)NCC1CC(NC(=O)CCc2ccnn2C)C1 c1(COC)cc(C(=O)NC2CCC2NC(C2CC(n3ccnc3)C2)=O)n[nH]1 c1(C(N(CC(C)O)CC#C)=O)ccc(CNC(=O)COCC2CC2)s1 N1(CC(C)NC(COC(C)C)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)CC1 N1(C(C(C=C)O)=O)CC(NC(=O)C=Cc2ncc[nH]2)CC1C C1(CNC(c2occ(C)c2)=O)CC2CC(C1)N(C(c1cnn(C)c1C(F)F)=O)C2 N1(CC(=O)NCC(CCN(C)C(c2cnn(C(F)(F)F)c2)=O)O)C(=O)CNC1=O Cc1cc(NC(=O)C(CCC2CC2)NC(c2c[nH]nc2C)=O)cc(CO)c1 c1(C(N(CCCNC(CC2C(OC)CC2)=O)C2CC2)=O)cc(C(N)=O)c[nH]1 C1(CNC(=O)CCOc2cccc(Br)c2)CC2(CC(NC(C3CC3F)=O)C2)C1 C1(NC(C=NOC)=O)CCCCCC1C(=O)NC(C)Cc1ccncc1 C=CC(C)(CCOC)C(=O)N1CC(NC(=O)CC2CC2C)C(C)(C)C1 c1(C(=O)NCC2CCN(C(c3[nH]nc(OC)c3Cl)=O)C2)cc2c(cc1N)OCO2 C1(NC(c2nn(CC)nc2C)=O)CC(O)CN(C(c2c(Cl)cnn2C)=O)C1 CCCCCC(=O)N(CC(N1CC=CC1COC)=O)C C(CC(=O)N(C)Cc1cocn1)(C(F)(F)F)NC(C(COC)(C)OC)=O N1(C(C2(NC(C3CC(F)(CF)C3)=O)C(C)(C)C2)=O)CC2(CCC(=O)N2)C1 c1(C(=O)NC2CCC(CNC(=O)COCC(F)F)C2)cnc2ccc(F)cc2c1 Cn1c(=O)c2c(ncn2CCC(=O)NCC2(CN)CC2)n(C)c1=O c1(C(N2CCC(O)(CC)C2)C(=O)Nc2cccc(OC)c2)ccc2ncnn2c1 C(C(=O)NCC1CCSC1)(C(C)(C)C)NC(c1ccn(COC)n1)=O N1(C(C(C)S(C)(=O)=O)=O)CCC2(CC1)CCN(C(=O)CC(C)C1CCCC1)C2 Cc1cccc(-c2cnc(CNC(=O)C(C)C(C)O)[nH]2)c1 C#Cc1cc(F)c(C(=O)N(C(CNC2CC(F)C2)C(C)(C)C)C2CCC2)c(F)c1 Cc1nnccc1C(=O)NC(CO)C(=O)N1CCC1C(=O)N(C)C C12(NC(CCc3cc(C)on3)=O)CCCCC1CN(C(=O)CCC(C)(F)F)C2 CC1SCCCC1C(=O)NC(C)C(=O)NCC1(CO)CCCO1 c1(C(N2CC(NC(c3ccc(OC)s3)=O)C3(C2)CC3)=O)cc(F)c(C)cc1Cl c1(CCC(=O)NC2C(NC(C(CC(=C)C)C)=O)CC2)ccc2c(c1)CCCO2 c1(O)cc(C#N)ccc1C.c1(O)ccccc1C=CC(=O)NCCCCCCCC CC1CCCc2nc(C(=O)NCC(CNC(C3(n4cnnn4)CC3)=O)CO)cn21 C#Cc1cccc(OCC(=O)NC(CNC(C2CC3CCC2C3)=O)CC)c1 Cc1cc(=NCC2CC(c3ccccc3)CO2)[nH]c(=NCc2cc(Cl)nc(Cl)c2)[nH]1 c1(C(N(C(CNC(COCCC=C)=O)C)C)=O)cc(N)cc(C(=O)OC)c1F c1(C(=O)NCC(C)NC(=O)CC2CCC(C)CO2)ncc(F)cc1F c1(CC)nc(C)c(C(N2CC=CC2CNC(=O)C(C(C)O)N(C)C)=O)o1 c1(CNC(C2C(COC)CC2)=O)ccc(O)nc1.N12CCC(C1)OCC2=O C1(C(=O)N(CCN(C)C(c2conc2C2CCCC2)=O)C2CC2)C(C(C)=O)C1(C)C C(c1ccc(O)c(O)c1)=CC(=O)NCCCCCN(C)C(C1CCCOC1)=O N1(C(C2CC(C#N)C2)=O)CCC2(CCCCN(C(C3CCCSC3)=O)C2)C1 N1(C(C2(C)CN(C(C3CCN(C)C3)=O)C2)=O)CC2COCC2(C)C1 Cc1sc(O)nc1C(N1CC2C(CNC(=O)CCOC(C)C)C2C1)=O CC(C(=O)NCC1C2CCCC12)C(C)S(C)(=O)=O C=CCN=C(NCCCOC(F)F)N1CCC(Oc2cccc(F)c2F)CC1 N1(C(C(C)(C)OC(c2n[nH]c3ccc(O)cc23)=O)=O)CCn2c(C(N)=O)cnc2C1 c1(OC)cc(F)c(C(=O)NC2CCN(C(c3nnn(C)c3N)=O)C(C)C2)c(Cl)c1 c1(C(=O)NC(C)CNC(c2ccc(C#N)s2)=O)cccc(F)c1Br C1(C(=O)NCC2(CC)CCCO2)CC2C=CC1N(C(=O)CNC(=O)OC)C2 c1(CC(N2CCCC(c3ncc[nH]3)C2)=O)c[nH]c2cccc(Cl)c12 C=C1COCCN(C(=O)C(c2cccs2)NC(=O)C(CCC)N(C)C)C1 N1(C(c2cccc(C)c2N)=O)CC(C)(C)CCC1CNC(=O)CCC(C)(C)F c1(C(N(C(C=C)C2CC2)C)=O)nc(CNC(=O)CSCC(F)F)oc1C C1(C(N(C2CCN(C)C2)C)=O)C(C2CC2)CCN1C(c1cc2cccn2cn1)=O CC(C)(C)CCCCC(=O)N1CCC2CCCC12C(=O)NCc1cnnc(O)c1 N1(C(CCc2c(C)cccc2)=O)CCC(NC(C2C3CCCC23)=O)C2(CCC2)C1 Cc1nc(C(F)(F)F)ccc1C(N1CC(=C(F)CNC(=O)C(C)(Cl)Cl)C1)=O c1(C(=O)NC2CC(NC(=O)COc3cn[nH]c3)C2)cncc(Cl)c1 C12(CC(N3C(C(C)NC(c4cn(CC)nc4)=O)CCC3)=O)CCC(CO1)C2 Cc1nn(C)c(C)c1CC(=O)NCCCN(C(C1CC2CC1C2)=O)C1CC1 C1(CNC(C2(CCOC)CCCC2)=O)CN(C(=O)Cc2cnoc2)C2CC12 CC(C(=O)NCC1CCN(C(C2CN3CCCC2C3)=O)CC1O)C(F)(F)F N#Cc1ccccc1-c1cn(CC2CN(C(C3CCC4CC3CO4)=O)C2)nn1 C1(C(N2C(C)CC(NC(C3(OC)CCCC3)=O)C2)=O)CN2CCN1C(C)C2 C1(C(N2CC(CN(C)C(C3CCCC3C(F)F)=O)C2)=O)Cc2ccccc2N1 c1(C(N2CC(C(C)NC(=O)Cc3cncs3)C2)=O)cc([N+](=O)[O-])n[nH]1 CC1CN(C(C2CNCC(C)O2)=O)c2ccccc2N1 C1(C(=O)NCC(C)CN(C)C)CN(C(c2coc(C3CC3)n2)=O)CCN1C C(=O)(C1=CSCCO1)N(CC(CC)NC(c1cccc(OC)c1F)=O)CC C(=O)(CN=S(C)(C)=O)N1CCN(CC(C)NC(C(CCOC)C)=O)CC1 c1(C(N2C3CCCN(C(C=COCC)=O)C3CC2)=O)ccc(S(C)(=O)=O)cc1F CCC(C)N(OC)C(=O)C1CC(NC(=O)C=Cc2ccncn2)C1 Cc1cc(NC(C2(C)CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)=O)c(C)cc1O C1(NC(CN(C2CCSC2)C)=O)(CNC(c2ncc(C(F)F)s2)=O)CCOC1 C(=O)(C(CO)C(C)(C)C)NCC(CNC(CC(C)(F)F)=O)C(F)(F)F N1(C(C(CCC)CC)=O)CC2CCN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2C1 C(=O)(C1CCc2c[nH]nc21)C(N1C2COCC1C2)=O.c1(CN)ccc(N)o1 N1(C(=O)CSC(F)F)CCCCC1c1cn(CC2CC3CC3C2)nn1 C1(CNC(C(C)OC)=O)C2CCCC1N(c1nc(C3CC3)nc(=N)[nH]1)C2 C(C(=O)NCc1cc(C(C)C)no1)(C(C)OC)NC(C=CC=CC)=O N1(C(C2CCCN(C(c3[nH]cc(C)n3)=O)CC2)=O)CCC(C)C(F)(F)CC1 C12(C(N(CC(CCC)O)C)=O)CCC(NC(c3cnc(C)nc3C)=O)(CC1)C2 N1(C(=O)C=CC2CCOC2)CC2CC(NC(C3CC(F)(CO)C3)=O)C2C1 CCCCC(CNC(=O)C(C)OC)NC(=O)CCCNC(C1CCC1C(F)F)=O c1(C(=O)NC2CCCN(C(C(C=C)O)=O)C2)ccn(CCO)c(=O)c1 S(=O)(=O)(c1ccc(NC(=O)Nc2c[nH]nc2C2CCOC2)cc1)N(C(CC)C)C c1(NC(=O)NC2CCC(CC(C)(C)C)C2)ccc(I)c(Cl)c1 c1(C(=O)OC)nnc(N2CC(O)(CCNC(C3CC3C(F)(F)F)=O)C2)s1 C1(C(N2CC(O)(CNC(c3cc4n(n3)CCCC4)=O)C2)=O)Cc2ccccc2S1 CCCCC(C)C(=O)N1CCSCC1CCNCc1cnc(OCC(F)F)cn1 C1(CNC(C(C)OCCC(C)C)=O)CCCCC1C(=O)NCCF C1(NC(C2(CCC=C)CN(C(c3cnns3)=O)C2)=O)CCC(C#N)CC1 C(C(C)N=c1cc[nH]cc1S(=O)(=O)NC1CCC(F)(F)C1)c1ncc(C)s1 C1(C(=O)NCCC(=C)CCNC(=O)CCNC(=O)CO)CC2CCC(C1)S2(=O)=O c1(C(=O)NCC(C)(CO)NC(CC(C)O)=O)cccc(N2CCCC2)n1 C(=O)(C(F)(F)C(F)F)NCC1(F)CC(NC(C2C(CC)CCO2)=O)C1 C(=O)(CC(C(F)(F)F)N(C)C1CC1)N1CCCC(CC=C)(NC(C2CSC2)=O)C1 N1(C(C(C)C(C)(F)F)=O)CCCC2(C1)CN(C(C1CC3(C1)CC(F)C3)=O)CCO2 C=CCC(CNC(c1cn2c(n1)CCC2)=O)C(=O)NC1CCCC2(C1)N=N2 N1(C(c2c(CC)c[nH]c2)=O)CCC(C)(CNC(=O)CC2CC2C2CC2)CC1 c1(SC)cc(C(=O)NC2CC(N(C(=O)COCc3ccnn3C)C)C2)ccc1F n1(C)cc(CCOCC)cn1.C12(SN)CC(C(=O)OC)(C1)C2 CCCC(CCC)C(=O)NC1CC1CNC(=O)CCNC(C1CCC1)=O Cn1[nH]c(=NC(=O)c2ccoc2NC(=O)C(C)(C)C)nc1N1CCOCC1 N1(C(CCC=C)=O)CCC2CN(C(=O)CC3CCCCN3C)CCC12 C1CN=C(NCC2CCC2(F)F)NC1.N1(C(C)=O)CCOCC1 C1(NC(Cc2ncc(C)s2)=O)CN(C(=O)Cc2cnoc2)CCC1C C1(CNC(c2cccc(C)c2)=O)CCCCC1N=c1cc(C)[nH]c(C)c1[N+](=O)[O-] CC1CC(C(=O)NCC2CC(F)(CNC(c3cn4ccnc4s3)=O)C2)=NO1 C1(NC(CC2ON=C(C)C2)=O)CCN(C(=O)C=Cc2ccncn2)CC(O)C1 Cc1cc(F)c(C(=O)N(C2CN(C(C3CCCC(C(C)(C)C)C3)=O)C2)C)c(F)c1 N1(C(C2(C#C)CCCC2)=O)CCC(N=c2nc(C(F)(F)F)[nH]s2)C(F)(F)CC1 N1(C(=O)C(c2nn[nH]n2)C2CC2)CCOC(c2nc[nH]n2)C1 N1(C(c2cccc(OCC=C(C)C)c2)=O)CCC(C)C(NC(c2cnc(O)s2)=O)C1 c1(NCC2(O)CN(C(c3c(O)ccc(OC)c3)=O)C2)nc(C)cc(C#N)n1 C1(OC)CCOC(CCNC(N2CCC(C(c3cccc(F)c3)=O)CC2)=O)C1 C(C(O)(CO)CO)NC(c1nc(CNC(C(C)OCCOC)=O)oc1)=O C1(NC(=O)Cc2cnccn2)CN(C(=O)CCc2ccc(F)cc2)C2CC12 CC(C)CC(O)C(=O)N(C)CC1CCN(C(=O)CSCc2ccccn2)C1 C1(CC(=O)N(C(C)C)CCN(C)C(C2C(C)(C)C2(C)C)=O)(CO)CCOCC1 N1(CC(C)N(C(C(=O)NCC(C)NC(=O)OC(C)(C)C)=O)C)CCCCC1 C(CS(=O)(=O)N=S(C)(=O)c1cn(C)cn1)(OC)OC(C)=O N1(C(CCCC)=O)CCC(C(C)(O)CNC(c2cc(C)n(C(C)C3CC3)n2)=O)CC1 C=CC(F)(F)C(=O)NCC1CC1NC(c1ccc(OCCN(C)C)nc1)=O C(=O)(CCCCC(N)=O)NCCSCC(=O)NC1(C)C(C)CCCC1 c1(C(N(C(c2cccs2)C)C)=O)coc(CNC(=O)C(N2CCOCC2)C)n1 CC(CN(C)C)CC(=O)N(CCCO)CCO.c12ccc-1s2 CCC(C(=O)OC)C(=O)NCCn1cc(C(=O)NCCn2cnc(CO)c2)nn1 c1(C(N2C(CNC(C3CC3(F)F)=O)CCCCC2)=O)csc2ccccc12 CCCCC(CN=c1[nH]c(C)ncc1C(=O)OC(n1cc(C(=O)NC)nc1)=O)NC C1(CNC(C2CCC(CC)C2)=O)CC(C)CN(C(C2(CO)CCC2)=O)C1 c1(C(=O)NCCC(=O)N(CC(C)NC(C2(C)CC(=C)C2)=O)C)ccccc1Cl N1(C(C2CC(O)(CC#C)C2)=O)CCCC(C)(NC(=O)C(=Cc2cccnc2)C)C1 c1(NC(=O)NC(c2cnn(C)c2)C)ccc2c(Cl)ccnc2n1 c1(C(=O)NCC(CCOC)NC(c2nnn(C)n2)=O)ccc(F)c2cnccc12 c1(CC)ncsc1C(=O)NC1(C(=O)NCc2ccsc2C)CCSC1 c1(C(C(=O)N(CCNC(C(C)O)=O)C)O)ccccc1C(F)(F)F N1(C(c2c(C)nc(C)[nH]2)=O)CCCCCC(NC(C2CCCC(C)(C)C2)=O)C1 C1(C(N2CCC(NC(C3(CC4CC4)CCC3)=O)C(O)C2)=O)CC2C=CC1CC2 N(C1CC(C)(C)c2ccc(Br)cc21)C(N1CCC(C)C1)=O c1(C(N2CCC(O)(CC(C)C)C2)C(=O)NCC(=C)C)nccc2ccccc12 C(CN=c1[nH]c(=NCCCCCCSC)c2[nH]ccc2[nH]1)c1nnc(CC)n1C C1(CN(C(c2cc(Cl)cs2)C(=O)NC)C)CC2COCC(C1)C2 Cc1cccc(C)c1OCC(=O)NC(C)CC(C)NC(C1CC1C#N)=O C1(C(=O)NCC2C(C(N)=O)C2)COCCN1C(=O)Cc1cnccn1 N1(CCC(N2CCC(C(C)NC(C34CC(F)(C3)C4)=O)C2)=O)CCSC(C)(C)C1 C(=O)(CCN(OC)C(=O)CNC(C1CC2CCCC2C1)=O)OCC c1(N2CCC(CCNC(c3cc(C(C)C)[nH]n3)=O)C2)c(C#N)cccc1[N+](=O)[O-] C1(C)(CNC(CN(S(CC)(=O)=O)C)=O)CCCC1NC(=O)CC1CCCO1 C1(CC(=O)NC(C(C)NC(c2cnc(-c3ccoc3)s2)=O)C)CCCCCC1 C1(c2nnnn2CC2CC2)(NCc2ccc(C(N)=O)cc2)CCC(C2CC2)C1 Cc1cc(C#N)cnc1C(N1CC(CNC(C23CC(C)(CO2)C3)=O)CC1C)=O Cn1ncnc1CN1CCC1(C)C(=O)NCC1CC1C1CC1 c1(C(C(=O)OCCCC)C)ccccc1-c1nncn1C C1(C(N2C(C(C)O)CC2)=O)(NC(=O)CC2COCC(C)O2)CCCC1C C1(C(=O)NCC2(NC(c3cn(CCCF)nn3)=O)CCC2)(OC)CCOCC1 Cc1c(C(=O)NCC2CCCC2NC(=O)CN2CC(C)C2)ccn1CCO C(=O)(CC(C(F)(F)F)NC(=O)C(CO)CO)NC(CCC)C(C)(C)C N1(C(C)C)CCC(N=c2nc(N(C)Cc3cnn[nH]3)c3ncn(C)c3[nH]2)CC1 CC1(C)Cc2cc(C(N3CCN(C(C4CSCN4C)=O)CC(O)C3)=O)ccc2O1 C1(F)(C(=O)NC(C2CC(F)(F)C2)CC)CCN(C(=O)OC(C)(C)C)C1 c1(NC(C(Cc2onc(C)n2)N)=O)ccc(Cl)cc1 CC(C)(C)CC(=O)N1CC(NC(=O)Cn2cc(Br)cn2)C(n2ccnn2)C1 c1(CCN2CCCC(C)(C(=O)OCF)C2)cccc2nsnc12 n1(CC(=O)NC(C(C)NC(=O)COC2CCC2)C)nnc(=N)[nH]1 C1(C2CCCO2)(C(=O)NCC2(O)CN(C(c3cc(Cl)cnn3)=O)C2)CCCO1 C1(CNC(=O)C(C2C3CCCC23)=O)COCCN1C(c1cc(Br)co1)=O c1(CNC(c2ccc(C3CCCCC3)cn2)=O)ccc(F)nc1 n1(CC(=O)N(CCC(C)NC(c2nccc(CC)c2)=O)C)ccc(=O)cc1C c1(NC(CC2(NC(=O)OC)CC2)=O)cc(C(=O)NCCc2ccsc2)n(C)n1 C1(CNC(C(C)OCCCC)=O)CC(O)CN1C(c1coc(C)c1)=O c1(OC)cc(C(=O)NCCCN(C(=O)C(C)(O)C2CCOC2)C)c2occc2c1 C1(CNC(C(C)O)=O)CN(C(c2cc(=O)cc(Cl)[nH]2)=O)CC1(C)C c1(C(=O)NC2C(NC(Cn3ccc(C)n3)=O)CC2)noc2c(F)cccc12 Cc1cc(C)c(NC(=O)CSc2cc3ccccc3s2)c(Cl)c1 n1(CC)c(C(N2CC(CNC(c3ccns3)=O)C(C)C2)=O)cc2ccccc12 Cc1ccnc(O)c1C(N1CC(N(C(=O)Cc2ccns2)C)C2(CC2)C1)=O N1(C(C)=O)CCC(O)C(C(=O)NCC2CC23CCN(S(=O)(=O)CCCCCl)C3)C1 C1(C(=O)NC2CC(CNC(c3ccc(C(N)=O)s3)=O)C2)CCCC2(CCC2)O1 CCC(CCC(=O)N1CCCC(C)(C(=O)NCc2cc(OC)ccn2)C1)OC c1(NC(C(N2CC(SCC)OCC2)=O)=O)nc2c(Br)c(C)ccc2s1 Cc1sc(Br)cc1C(=O)N(C(C)CNC(=O)C(c1ccc(O)cc1)=O)C Cc1ncc[nH]c1=NCc1cc(Br)ccn1 C12(CNC(C3C(COC)C3)=O)CC1CN(C(=O)COCCc1ccccc1)C2 C#CC1(C(=O)NCC(C)(COC)CC)CCN(C(=O)C(C)CC2CCC2)C1 N(C1COc2cccc(C)c21)C(C(N1CCCC(CCOC)C1)=O)=O N1(CC(=O)NC(C(C)NC(C2C(C(=O)OC)CC2)=O)C)CCCC1C Cc1nc(C(C)C)cc(=NCC2CC(CNC(=O)C3=CCCCCC3)CO2)[nH]1 C1(CC)CCOCCN1C(C1COCC1NC(c1n[nH]c2c1CCC2)=O)=O C(=O)(CC1COCc2ccccc21)NC1CCC(NC(c2c(C)nsc2)=O)CC1 c1(CC(N2C(CN(C(c3c(C)nc(CO)s3)=O)C)CCC2)=O)cccc(Cl)c1F c1(CCNC(=O)NC2CC3C=CC2CC3)c[nH]c2ccc(Br)cc12 c1(C(N2C(CC(N3CCCC(C#C)C3)=O)CCC2)=O)nn(C)c2ccccc12 N1(C(C)=O)CCCC1C1CCCC1.NS(=O)(=O)NCCNC(=O)CC1CC1.C12CC1C2 c1(OC)c(C(=O)NCCCCC2CN(C(c3cc(C)oc3C)=O)C2)sc(Cl)c1Cl C1(C(N2CCC(F)C(F)C2)=O)N(C(=O)C2=COCC2)CC12CCCC2 C(CN=c1[nH]n2cc(C)nc2s1)NC(N1CCCC(CC#C)C1)=O Cc1c(C(=O)NCC2CCC2NC(c2cccnc2C(F)F)=O)cncc1Cl C1(C)(NC(C(CSCC)NC(c2cnc(CC)[nH]2)=O)=O)CCCOC1 C(C(C)(CC)C(=O)NCCS(=O)(=O)CC)NC(CC)=O O=C(C(O)CC(F)(F)F)NCCCNC(C1CC1C(F)(F)F)=O c1(C(N2CC(OC)C(NC(=O)CCNC(=O)CC(C)C)C2)=O)ccc(F)cc1N c1(C(=O)NC2CCCN(C(C(C)=C3CC3)=O)CC2F)ccc(S(N)(=O)=O)c(C)c1 CC(C)P(=O)(CC(=O)NCC1CC1NC(c1cn(C)cn1)=O)C(C)C c1(C(=O)NCC(CNC(C2CC(OCC)C2)=O)O)cnn(-c2ccccc2)c1Cl N1(C(CCN(C(CC)CC)C)=O)CCC(NC(c2[nH]cnc2C)=O)C1 c1(C(N2CCC23CCCC3)C(=O)NC2CC(F)(F)C2)cc2ccccc2cn1 C(=O)(C1=C(C)OCC1)NCCN(C(C1CCC(OC)CC1)=O)CC1CC1 c1(C(=O)NC2CCCC(NC(CCc3nc(C)sc3)=O)C2)ccn2nccc2n1 c1(C(N(CC(C)NC(CCN(CC)CC)=O)C)=O)cc(C)c(F)cc1N CCCC(CNC(=O)Cc1ccnn1CC)NC(c1cc(CC2CC2)[nH]n1)=O.OC C1(NC(CCCNC(C)=O)=O)CC2C(NC(=O)C=CCF)C2C1 C1(CC)(NC(=O)COc2cc(C)on2)CCCN(C(c2cncc(SC)c2)=O)C1 C1(NC(Cc2cc(C)on2)=O)CN(C(=O)CCC2CCCCN2C)CC1CO C1(NC(c2cc(OC)cc(Cl)c2)=O)CC2CCC(C1C)N2C(=O)CC(F)(F)F C(=O)(C1=CC(O)C(NC(=O)COC2CCCOC2)C1)NC1OCCC(C)(F)C1 C1(CNC(=O)Cc2csc(Br)n2)CCC2(CN(C(C3(CF)CCC3)=O)C2)O1 N1(CC(=O)NC2CCC(CCC(=O)NCCSC(C)C)C2)CCOC1=O N1(C(COCC(=O)NC)=O)CC(CNC(=O)Cc2cccn2C)C2CC12 C1(CC(N2C(CC)C(NC(=O)C(C)(C)SC)CC2)=O)CCCC(C)(C)C1 C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C)CCN(C)C(C1CC2CSCC(C1)C2)=O c1(C(N2CCC(CCNC(C(CC)CO)=O)C2)=O)ccc(C)nc1C c1(C(N(C2CN(C(C(C)CF)=O)C2)C)=O)cc(C(C)C)oc1C(C)C c1(Cc2nc(-c3cccc(C)c3)nn2CCCCO)ccc(Cl)c2cccnc12 N1(C(=O)Nc2c(CC)nn(C)c2)CCC(C)C(CNC(=O)C(O)P(C)(C)=O)C1 N1(C(C(CCOC)NC(=O)CC2CCCSC2)=O)CCC2C(OC)CC12 N1(C(COCCCOC)=O)CCCC(C)(CNC(C2(C)CC2(F)F)=O)C1 Cc1ccc(F)c(CNC(=O)CC23CCC2CN(C(C2CCCOCC2)=O)C3)c1 C1(CCC)CCN(C(C2(CNC(=O)C(C)n3ccnn3)CC3(CC3)C2)=O)C1 C(=O)(CCC(=O)NC(Cc1ccccc1Br)C(=O)NCCN(C)C)NCC N1(CC(C)NC(c2cnc(CN)s2)=O)CCN(C(c2ccn(C3CC3)n2)=O)CC1 C#CCCCC(C)C(=O)NC(C)(C)C(=O)NC1CC(O)C(O)C1 C12(NC(CCCC#C)=O)CCCN(C(=O)CCC(C)C)CC1C2 N1(C(C=CC=CCC)=O)CCOC2(CCC(NC(C3CCC(=O)O3)=O)CC2)C1 C=C(Cl)CCC(=O)NC(CCSC)C(=O)NCCN1CCCCC1C C1(NC(CCN2CCN(C)CC2)=O)CCN(C(c2cccc(N)c2Cl)=O)CC1F c1(C(N(C2CCN(c3cc(OCC=C)ncn3)C2)C)=O)ccnc2ccccc12 Cc1nc(CC(F)(F)F)sc1CC(=O)NC1CC1NC(c1cnsn1)=O c1(CCN(C)CCN(C(c2cn(C3CC3)nn2)=O)C2CC2)ccc(=N)[nH]c1 c1(C(=O)NC(CNC(C=CCOC)=O)C(C)C)cncc(-n2cnnn2)c1 c1(C(N2C(C(N3C(C(C)C)COCC3)=O)CC3CC32)=O)cccc2ncccc12 N1(C(COCCCC)=O)CCC2(CC1)CCN(C(c1c(C)oc(C)c1C)=O)C2 Cc1ccc(OCC(N2CC(N(C(=O)C(c3ccccc3)C)C)C2)=O)c(Br)c1 C(=O)(C(C)(C)C1=CCN(C(=O)CN(C2CCC2)C)C1)N1CCCC(=C)C1 CC(C)C(C)C(C)NC(=O)CC1(N(C)C(c2cccnc2O)=O)CC1 C#Cc1ccc(C(=O)NC2CCC2CNC(C2(C(C)C)CC2C(F)(F)F)=O)nc1 Cc1c(Cl)ccnc1C(=O)NC1CN(C(=O)CC(=O)N(C)C)CC1O S(=O)(=O)(CCCCCl)NC1C=CC(C(=O)NC2(c3ccn(C)n3)CC2)C1 C1(C2CN(C(=O)Cn3cc(Br)cn3)C2)(NC(c2ccc(C(C)=O)cc2)=O)CC1 N1(S(c2cnn(C(C)C)n2)(=O)=O)CC2CCCC(O)C2C1.C12CCCC1CC2 Cc1ccnc(O)c1CNC(=O)NC1CCCCC1(F)F c1(C(=O)NCCN(C(C2C(CC)OCC2)=O)CC)ccccc1-c1cn[nH]c1 C(C1CCc2ccccc21)Nc1cc(N(C)CC2CCC(=O)NC2=O)ncn1 CCCCCC(C)CC(=O)N(CCCN(C)C)CCNC(c1cccc(CO)c1)=O C(=O)(C(C)NC(=O)CCSC(C)C)NC(COCC)C c1(CN2C(C)C(NC(=O)CC3(CO)CC3)CCC2)ccc2c(c1)OCCCO2 C1(NC(Cc2nc(C)sc2Cl)=O)CN(C(C2CCOCC2)=O)CCC1F C=CCCC(C(=O)N(CCC(C(C)C)NC(=O)CCCC)C)c1ccccc1 N1(C(C2CN(C3CC3)CCS2(=O)=O)=O)CCC2CCC(C1)N2CC1CCCC1 C(CC(F)(F)F)N(C(C1(CNC(c2ccc(CO)o2)=O)CCCO1)=O)CC Cc1nc2nccc(N3CCC(CNC(=O)NC4CCc5ccnn5C4)C3)n2n1 N1(C(C(C(C)O)(F)F)=O)CC2CCN(C(=O)CCSc3ccncc3)CCC2C1 N1(C(C2(O)CCC2)=O)CC(NC(C2(c3ccccc3)CCC2)=O)CC1CO N1(C(C(C(=O)OCC)C2CC2)=O)CCN(C(=O)COCCSC)C2COCC12 c1(-c2nccc(-c3n(CC(C)(C)NC)ccn3)c2)c(C)nn(C2CCOC2)c1C c1(C(=O)NCC(CC)NC(c2c(C)ncn2C)=O)cccc(Br)c1N C1(C(=O)NCC2N(C(C3CCC(C)CC3)=O)CCC2C)CC2(CCOC2)C1 C(C(C)(C)C(=O)NCC(O)CNC(C1CCC(=O)NC1)=O)OC(C)C C1(C2CCOCC2)(CNC(=O)Cc2cncnc2O)CCN(C(=O)CCF)C1 c1(OCC)ccc(F)c(CNC(=O)C(N2CCN(CC)CC2)c2cn[nH]c2)c1 C(=O)(C1=CC(C)(C)C1)NCCCCC1N(C(=O)CCC(=O)NCCC)CCC1 Cc1ncc(CC(=O)NC(C2CCN(C(c3nc4c(s3)CCC4)=O)C2)C)c(O)n1 c1(C(N2CCN(c3ncc(F)cn3)CC2)C(=O)NCCC)c(Cl)nc(Cl)n1C C1(CNC(=O)C#CC2CC2)CC2(CO1)CN(C(=O)Cn1cnc(Br)n1)C2 c1(C(=O)NCCN(C(=O)CSc2ccccn2)CC)cccc(Cl)c1F C1(CNC(c2cncc(NC)c2)=O)CCN(C(c2cc(C)cc(F)c2)=O)C(C)C1 c1(C(N)=O)cc(C(N2CCC(CNC(=O)CCN3CCOC3=O)CC2)=O)ccn1 C1(N(C)C(c2ccc(=O)oc2)=O)CN(C(C2CCOC(=O)N2)=O)CC1O c1(OCC)ccccc1CCC(=O)NCC(C)N(C)C(c1cnn(C)c1)=O N1(C(CCc2cnc(C)s2)=O)CC(NC(=O)C(F)(F)c2cnccn2)C(O)C1 Cn1ccc(=O)c(C(=O)NCC2CC(F)(CNC(C3CCCOCC3)=O)C2)c1 N1(C(C2C(OCC)C2)=O)CCN(C(c2c(Cl)n[nH]c2CC)=O)CC(C)(C)C1 C1(CCC(=O)NC(C)CC2CCC2)CCCN(C(=O)CC2CNC(=O)O2)C1 CCCC(C(=O)NC(C(=O)NC1C2COCC12)C1CCC1)OC C1(NC(C(C2CCCOC2)OCC)=O)CCN(C(=O)CCOCCOCC)C1 c1(C(=O)NC2CN(C(=O)CCc3cccc(Br)c3)C2)cc2cccc(Cl)c2[nH]1 N1(C(=O)NC2CC(c3ccncc3)C2)CCC2(CCC(O)C2)C1 C#CC(CNC(=O)CC1(OC)CN(C(c2cnc(Cl)s2)=O)C1)CC C(C(F)C(=O)Nc1cn(C(c2ccccn2)C)nn1)C1CN(C(C)=O)C1 c1(C(=O)NC(CN(C(=O)C=C2CCC2)CC)C)cncc(OCC(F)(F)F)c1 C1(c2n(CC3C(C)C3)nnn2)(NC2COC3(CCC3)C2)CCCSCC1 C1(N(C(C(=O)OC)=O)C)CCN(C)CC1.N12CCC(C1)OCC2=O C(C(O)CC(=O)NCCCC(F)F)NC(C(CC)OC)=O c1(C(=O)NCC2C(C)CCN(C(CC=C(C)C)=O)C2)ccc2nc(C)[nH]c2c1 CC#CC1CN(C(C2CCCCC2CNC(c2occc2C2CC2)=O)=O)C1 C(=O)(CC1NC(=O)c2ccccc21)N(C1CN(C(=O)Cc2cnns2)C1)C c1(C(=O)NC2(CNC(CNc3nccc(OC)n3)=O)CC2)ccc2cc(C)oc2c1 Cc1ccccc1OCC(N1CCCC1CCNC(=O)CCc1nccn1C)=O C1(C(C2CCC2)OC)CCC2(CC2)N1C1(CO)CN(CC2CCCCCC2)C1 c1(C(=O)NCCC(N2CCN(C(C)=O)CC2)=O)cc2ccccc2[nH]1 C(=O)(C1=CCC2(COC2)OC1)N1CCN(C(c2c(C)n3c(s2)ncc3)=O)CC1C C1(NC(C(C2CCC2)OC)=O)CN(C(=O)CSCC(F)(F)F)CC1C c1(C(=O)NCC(C)(O)CNC(C2CC(C(F)F)C2)=O)cnc2ccccn12 c1(OC)cc(C(=O)NCCN(CCOCCO)C(CC(C)C)=O)on1.C1(S)CC1 C#Cc1cccc(C(=O)NC2CCCCCN(C(=O)Cc3ncc(C)[nH]3)C2)c1F c1(C(N2C3(C(=O)NC4CCOCC4O)CC(C2)C3)=O)ccc2c(c1)CC2 Cc1cn2c(C(=O)NC(C)CN(C)C(C3(CCF)CC3)=O)c(Cl)nc2s1 N1(C(=O)OC(C)(C)C)CCC2(CC1)CC(C(=O)Nc1cnc3scnc3c1)CCO2 C(C(C(=O)NC)C(C)C)NC(c1c(CC)ncs1)=O.C12CC(C1)OC(=O)N2 N1(C(c2c(CC)cncc2)=O)CCC(C)N(C(c2nn(C)cc2[N+](=O)[O-])=O)CC1 C12(O)CCN(CC1)C2=O.N1(Cc2cccc(OC)c2)CC2CC(O)C2C1 c1(C(=O)NC(C)CCCNC(C2CCC3CC2CO3)=O)cc2cc(Cl)cnc2[nH]1 N1(CC(C)(C)OCC)CCCC(CCN(C)CCO)C1 C=C(C)CC(C(=O)N1CCC(C(=O)NCCCc2ncn(C)n2)(CO)C1)OC C(C(CC(C)C)C(=O)N(CC(=O)NC1CC1)C)NC(C(CCC)OCC)=O C1(NC(C2(C)CCC(=O)N2)=O)C2CCC1CN(Cc1ccc(-c3cccs3)o1)C2 C1(C(=O)NC(C(C)C)CNC(=O)CC(C)C2CC2)CCC(=O)C1C Cc1c(C(N2CC(C)(NC(C3COC(C)C3)=O)C2)=O)cnn1-c1ccc(F)cc1 C(C(C)(C)C(=O)N1CCC(Nc2cc(NC)ncn2)C1)SC C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1C(CNC(c2ccc(OC)cn2)=O)C1 Cc1c(C(N2CC(CNC(C3CCCC3O)=O)C2)=O)cc(C)c2ncccc12 CC(C)C(CNC(C1(CF)CC1)=O)NC(=O)COC1CCOC1 c1(-c2cn(C)nn2)ncccc1C#N.Cc1ccc(CCC(=O)N2CCC2)o1 C1(C)(C(N2C(C)(CNC(CS(CC)=O)=O)CCC2)=O)CC(C2CC2)=NO1 C#CCCC(O)C(=O)N1CCCC(N(C)C(c2csc(C)c2)=O)C1 C1(F)(CNC(c2c(CC)c[nH]n2)=O)CCC(CNC(c2ccc(=O)n(C)n2)=O)C1 N1(C(c2c(C(C)C)c[nH]n2)=O)C2CCC1C(CNC(C1CC3(CCO1)CC3)=O)C2 C1(C(=O)OCC)COC2(C(N3CC(OC)C(OC)C3)=O)CC1C2 c1(C(=O)NCc2ccc(-c3n(CC)nc(C)c3)cc2)c(F)ccc(C)c1Cl N1(C(c2cc(C)cc(Cl)c2)=O)Cc2ccccc2CC1C(=O)NC1CN(C)C1 CC#CCCCC(=O)N1CCC(C(=O)NCC2(C)CSC(C)=N2)C1(C)C c1(OCC)ccc2c(c1)OCC(C(=O)N1CC(F)(F)C1C1CC1)=C2 CN1CCOCC1CC(=O)NC1CC(NC(=O)CC2CSCCO2)CC1O C1(C#N)(Cc2n(-c3ccn(CC)n3)nc(CS(C)(=O)=O)n2)CC(C)(C)C1 CC1CC(=O)NC(C(N2CC3CC2CN3C(C2(C(=O)N(C)C)CC2)=O)=O)C1 C1(O)(C(N2CCC(CNC(C(C)SCC)=O)CC2)=O)CCCCCC1 C1(NC(c2cnc(C)nc2O)=O)CCN(C(=O)CCC(F)F)CCC1CO N1(C(C2(C)CC2)=O)CCCCC(CNC(=O)C(O)COCc2ccccc2)C1 c1(CC(N2CC(NC(c3c(OC)nn(C)c3)=O)C3C2C3)=O)ccc(O)cc1Cl C12(C(N3CC(C(N4CCC(OCC=C)C4)=O)OCC3)=O)CCCC1CCC2 N1(C(C(=O)NC2CCC(CCCCCC)CC2)=O)CC2(C)C(=O)NC(=O)C2(C)C1 N1(C(c2c(C)sc(Br)n2)=O)CC2CC(NC(=O)CCCC3CC3)C1C2 Cc1nc2c(cc1C(=O)NC(c1cn(CC3CC3)nn1)C)c(C)nn2C C(=O)(C(CC(C)C)NC(=O)C(C)CNC(N)=O)NC(C(=O)OC)(C)CO C1(CNC=O)CCCCCC1NC(=O)CNC(=O)N(C)C.c1scnc1C(C)(C)C C1(C(=O)NC2(CCC=C)CC2)CCCN(C(=O)C(C2CCCCC2)F)C1 CC1COCC(C(=O)NC(C2CCCCC2)C(=O)NCc2cc(O)ncn2)O1 C1(C(=O)NCC(C(=O)NC(CC=C)CC)C)CC2(CCO1)CC2 C1(C(=O)NC2CC(C(C(=O)NCC(CO)OCC)F)C2)CC1C1(C)COC1 N12CCC(C(C)C1)C2.Cc1cccc(OCCNC(=O)CC(C)C)c1 Cc1cc(=O)c(C(=O)NCC2(F)CN(C(=O)C3=C(Cl)CCC3)C2)cn1C1CC1 C1C(C)(CN(C)C)C(=O)O1.n1(C(C)C)cc(C(O)CCO)nn1 c1(C(N2CCC(NC(CCOCCCOC)=O)CC2C)=O)cc(Cl)c(Cl)cc1C c1(CC(=O)NC(CC)CNC(=O)CCSc2cccc(Cl)c2)cc(Cl)n(C)n1 Cc1ccc(C=CC(N2CC=CC2(C)C(=O)NCCSC(C)C)=O)cc1 C1(CNC(c2ccc(C)cc2F)=O)CN(C(C2(F)CCOC2)=O)CCC1(C)C N1(C(C2OCCN(CC)C2)=O)CCC(CNC(C2(O)COC2)=O)CC1C c1(C(=O)Nc2nc(-c3c(C)cnc(F)c3)sc2)cccc2cn(C)nc12 n1(CC)cc(Br)cc1C(=O)NCC1CC(NC(=O)Cc2ccc(Cl)cc2)C1 C(=O)(C(O)CCNC(=O)CNC=O)N(CCC(C)NCCC#N)CC N=c1nc(C(=O)NCC2CCN2C(c2csc(Cl)c2Br)=O)cc[nH]1 C12(C(N3CCCN(C(C4C(C=C)CC4)=O)CC3)=O)CC3CC(CC(C3)C1)C2 CCC(C)CC(C(=O)N1CCC(NC(N)=O)C1)NC(c1ccns1)=O Cc1cnc(NCCCC#N)c(S(=O)(=O)NC(c2cnns2)C)c1 C(=O)(CN=c1cc[nH]cc1)N1CCC(NC(COCCC=C)=O)(CC)CC1 C1(NC(C=C(CCC)CCC)=O)COC2(CCN(C(C3CC3(Cl)Cl)=O)CC2)C1 c1(OCCCNC(CN2CC(C)C2)=O)ccccc1.C1(=O)C(C)C2CC12.C1CNO1.O CC(C(=O)N(C1CC(NC(C2CCOC2)=O)C1)CCO)C(=O)N1CCOCC1 c1(CCCNC(N2C(C)CSCCC2)=O)cc(F)c(F)cc1F N1(C(C(COC)COC)=O)CC2(CNC(=O)CCc3ccc(C)cc3)CCC1C2 Cc1nc(C(=O)NC(C(=O)NCC2CCCCCC2)C2(C)CC2)sc1C c1(C(N2CC3(C2)CN(C(C2(F)C4CCCCC24)=O)C3)=O)cc2n(n1)CCOC2 C(=O)(C(C)(C#N)CC)N1CCC(CC(=O)N(C)Cc2c(CC)cccc2)C1 C1(CNC(C2CC(F)C2)=O)C2CN(C(c3sc(Br)cc3F)=O)CC12 C1(OC)COCCC1NC(c1c[nH]nc1CNC(C1CCC2CC12)=O)=O C(C(F)(F)C(=O)N1CCC(C(C)CNC(c2ncccc2F)=O)CC1)OC Cc1nnc2n1CCCC2C(=O)NCC1CC(NC(=O)CCCC2CCCO2)C1 C(C1=C(C#N)CCC1)NC(C1CC(c2ccccc2)C1)C CC1C(NC(c2cc(O)n(C)n2)=O)CC2CCC1N2C(C1(S(N)(=O)=O)CC1)=O c1(C(N2CC(C(C(=O)N(C3CCCC(C)C3)C)SC)C2)=O)ccc2ccoc2c1 CC1(CNC(c2cscc2Cl)=O)CCCN(C(c2ncnc(O)c2F)=O)C1 N12Cc3cccc(c3C1)C(=O)NN(C(C(C)C)=O)CC2=O.C1(CC)CCOC(C)C1 c1(C(=O)OC(C)C(=O)N(C2CCCCC2)CC(c2cccs2)O)ccccc1C#N c1(OC)cccc(C(N2CCCC2CSC2CC2)C(=O)NCc2nccs2)c1Cl C1(NC(CCCCC(C)C)=O)CCN(C(c2nccc(C#N)n2)=O)C12CCCC2 C1(NC(CC2C(C)(C)C2)=O)CC(C(=O)NC2CCC3(CCC3)C2)C12CCC2 C12(C(NNC(c3c(N)cc(Br)cc3)=O)=O)CCCC(C1)C(=O)NC2 N1(c2n(C(C)C)c(-c3c4c(nn3C)CCCC4)nn2)CCc2nccc(N)c2C1 c1(COCC)[nH]c(C2CCN(C(=O)OCS)CC2)cc1C.C123CC(C1C2)N(C)C3=O N#Cc1ccc(SCC(N2CCC(N3CCC3)CC2)=O)cc1.C12CC(C1)C(=O)N2 Cc1cc(=NC(=O)C(=O)N2CCCC2CNC(c2cccc(F)c2C#N)=O)[nH]o1 C(=O)(CS(=O)(=O)C1CCCC1)NCC1CN(C(C(CC=CC)C)=O)CC1(C)C c1(C(N2CCC(F)(CNC(C3CC34CCC4)=O)C2)=O)c(F)cc(C2CC2)cc1F N(C1CCC(NCC(c2cc(C(C)C)nn2C)=O)c2ccccc21)C(=O)OC(C)=O c1(CCCC)ccc(C(N2CC(CNC(=O)C(F)=C(C)C)C3CC23)=O)cc1 N1(C(CCN(C(C)=O)C)=O)CCC2CCN(C(=O)CC(C)F)CC12 c1(C(=O)NC2C(CNC(=O)COCC3CC3)CCC2)coc2c1CS(=O)(=O)C2 N1(C(CN2CC(CC)C2)=O)CCC(NC(=O)CCc2cncs2)C(O)C1 C(C(=O)N1CC(CNC(c2n[nH]c(C)n2)=O)C1)(C(C)C)OCC c1(C2(C(=O)NC(C)CN(C)C(C3CC(C)(F)C3)=O)CC2)ccc2c(c1)OCCO2 c1(CC)ncccc1C(=O)NC(CC(=O)NCCC1CCCCO1)C1CC1 c1(CC)nc(C)oc1C(=O)NCCOC(C)(C)CNC(C1CC2(CCC2)C1)=O C(=O)(C(F)C(C)(F)F)N1CCCC(C(=O)NCc2cc(OC)no2)C1 C1=CC2CCC1C1CN(N3CCC(c4ccccc4)CC3)CC21 C(=O)(CC(C(=O)NC(C1(CC(c2ccc(C)o2)=O)CC1)C)NC(=O)C1CC1)OC Cc1cccnc1CCC(=O)NC1CN(C(C2CC3(CCC3)C2)=O)CC1F CC(F)CC(=O)NCC1(O)CN(C(=O)C=CC(c2ccccc2)=O)C1 C1(C(C)C)(CO)CCCN(C(c2cnc(C(F)(F)F)s2)=O)C1.c12cc(ncn1)CN2 N1(C(c2c(OC)csc2)=O)CC2CN(C(c3ccc(Br)c(OC)c3)=O)CC12 Cn1cc(C(=O)NC23CC2CN(C(C2CCC(CC(F)(F)F)CC2)=O)C3)nc1O C12(CNC(C(C)OCCCC)=O)CN(C(c3c(C)ncn3O)=O)CC1CCO2 C1(N(C)C)CN(C(=O)NC(C)CC(O)c2ccco2)C2(CCCC2)C1 N(C(=NCc1cccc(F)c1)N1CCC(c2cc(C)cc(C)c2)C1)CCSC C(CC(C)(C)C#N)(c1n(CC(=C)C)nnn1)NCCc1ccc(Cl)cc1 c1(C(=O)NCCOCCNC(=O)COC(F)(F)F)cnc(O)c([N+](=O)[O-])c1 c1(C(N2CC(CC(=O)NCCCc3cncnc3)C2)=O)cc(O)cc(O)c1 c1(OC)c(C(N2CCSCC2CCNC(C23CC(F)(C2)C3)=O)=O)ncnc1C c1(-c2ccc(CNc3cccc(NC(C)=O)c3F)nn2)cc(F)cc([N+](=O)[O-])c1 c1(CC)oncc1C(=O)NCC(O)CNC(c1ccc(C(=O)NC)[nH]1)=O Clc1cc(NCCCN2CCN(c3cc(Br)ccn3)CC2)ccc1Cl N1(C(C#CC(C)(C)C)=O)CC2CC1CN(C(c1c(Cl)cnn1C1CCCC1)=O)C2 c1(OC(C)C(=O)NC2(C)CC(C(=O)O)CS2)ccc(-c2nn[nH]n2)cc1 N1(C(C2CN(C(C)(C)C)C(=O)C2)=O)CCC2(C1)CN(C(=O)C#CC1CCCO1)C2 C1(CNC(c2ccc(O)cn2)=O)CCCCN(C(=O)Cc2ccccc2Br)C1 C1(NC(C(F)=CC)=O)CN(C(C2CC(=O)N(CCN3CCCC3)C2)=O)CC12CC2 C1(N(C(COCCCOC)=O)C)CCCN(C(=O)Cc2c(C)cnn2C)CC1 c1(C(N2CCC(CNC(C(CCC)C(C)C)=O)C2)=O)cnc2[nH]c(C)nc2c1 CCC(C(=O)NCC1CC1NC(c1csc(CCP(C)(C)=O)n1)=O)C(F)(F)F N1(C(COC(CC)C)=O)CC2CC(C1)CN(C(C1(c3ccncc3)CC1)=O)C2 N1(C(C(CC(C)C)=O)=O)CCCCCCC1C(=O)NCC1(CN(C)C)CCC1 c1(C(N(CCSC)CC)=O)ccc(NC(=O)C(C2CCCO2)OC(F)F)cc1 Cc1ncccc1CC(=O)NC(CC1CCCC1)C(=O)NC1CC(C#N)C1 C12(C(N3CC(C)(O)C3)=O)C(NC(c3ccc(C#N)[nH]3)=O)C3CC1C2C3 C1(N(C)C(c2cc([N+](=O)[O-])co2)=O)CNC(=O)CN1Cc1ccccc1 CS(=O)(=O)C1CC(C(N2CC3(CCC3NC(=O)Cn3ncccc3=O)C2)=O)C1 C1(NC(=O)NC(CCN2CCCCC2)C(=O)O)CCCC2(CC1)CC2 O=C1CCCC(C(=O)NC2CC(O)C2CC(=O)NCc2ncc[nH]2)CC1 C#Cc1cccc(CNC(=O)NC2CCN(C3CCC3)C2=O)c1 C(CCCC(=O)NC(CCC1CC1)C(=O)NCc1cc(O)ccc1C)(OC)OC CC(C)C(C)(O)C(=O)NCC1(CNC(C2(c3ccc(F)cc3)CC2(C)C)=O)CC1 c1(C(N2C(CNC(C=NOC)=O)CC(O)C2)=O)c[nH]c2ccc(F)cc12 c1(N2CCC(NS(NC)(=O)=O)CC2)nc(=N)[nH]c(=NCCN2CCC(C)CC2)[nH]1 c1(CCC(N2CCCC(CNC(C(C)S(C)(=O)=O)=O)C2)=O)nc2cccnc2[nH]1 N1(C(c2cncc(CNC(Cc3c(C)nsc3)=O)c2)=O)CCC12CCCCC2 CC(C)(C)C#CC(=O)NCC1CC(F)(CNC(=O)C(C)(C)c2ccccn2)C1 C1(CNC(C(CCOC)C)=O)CN(C(c2ccc(N)cc2F)=O)CCCO1 c1(OC)ccc(F)c(OC(CC(c2ccc(CC3CC3)c(F)c2)(F)F)=O)c1 c1(CCCC)cc(C(=O)N(C(C)CNC(=O)C=Cc2c[nH]nc2C)C)c(C)o1 N1(C(CCNC(COC)=O)=O)CCN(C(=O)C#CC(C)(C)C)C(C(C)C)C1 C1(CS(=O)(=O)NC(CC)CN2CCCC2)CCC12CCC2 c1(C(=O)NCCCN(C(C(C)CC2CC2)=O)C)ccnc(O)c1 C1(C(=O)NC23CC(NC(=O)Cc4ccccc4F)(C2)C3)CCC(C2CC2)C1 c1(C(N(c2nnn(C)n2)Cc2c(F)ccc(F)c2Br)=O)ccc(S(C)=O)c(F)c1 C1(CNC(CCCCC=C)=O)CC(C)CN(C(C)=O)C1.C(=O)(C(F)CN(CC)CC)N CCCCC(CC(=O)NCCCNC(C)=O)NC(=O)C(COC)OC CC(=O)CCCC(C)C(=O)N1CC(C(=O)N2CC3(CC3)C2)c2ccccc21 c1(CCC)nc(C(=O)NCCCCCN(C)C(C23CC(C(C)C)(C2)C3)=O)co1 C(=O)(C(C)(C)Cc1cnn[nH]1)NCCN(C(=O)C(C)CCN(C)C)CC c1(NC(=O)NCC2C(c3cccc(OC)c3)C2)nccc(OC)c1F c1(OC)c(Br)ccc(CN2CCC(OCC3CCCCC3)CC2)c1F Cc1nccnc1C(=O)NC1CCCCC1NC(=O)C(C)(C)OCC(F)(F)F N1(C(CNCCCC(C)C)=O)CCN(C(=O)OC(C)(C)C)C(CS(C)(=O)=O)C1 c1(-c2cn(CCCCCCNC(CC(C3CC3)OC)=O)nn2)cc(C)cc(Br)c1 C(C(=O)N1CCC1CNC(c1cccc(-n2cccn2)c1)=O)(C(C)C)OC CCCCC(F)C(=O)N(CC(O)CNC(=O)C(CO)N(C)C)C C1(NC(C(C2(C)CC2)NC(=O)CCc2ncc[nH]2)=O)CCOC1=O C1(CNC(c2cc(CC)oc2C)=O)CN(C)CCN1C(=O)Cn1cnnn1 C(C(=O)NCC(C)NC(c1ccc(CC)cc1)=O)(C(C)C)SCC N1(C(Cn2nnc(C)n2)=O)CCCN(C(=O)CSS(C)(=O)=O)C(C)C1 Cc1cc(C(=O)NC(C2CN(C(c3c(C)noc3C)=O)C2)C)c(C(F)(F)F)o1 c1(CNC(c2c(C)nc(O)[nH]2)=O)nnc2n1CCN(C(C1CCCN1N=O)=O)C2 CC(C)CC(C(=O)NCC12CC(NC(c3cncc(F)c3)=O)(C1)C2)C(N)=O C(=O)(C(CC(C)C)C(C)C)NCc1cc(C)c(NC(=O)C(F)(F)C(C)(C)O)o1 Cc1ccc2c(c1)CC(C(=O)NC1CCC1NC(c1c(C)nc(=N)[nH]c1C)=O)O2 CC1(C)CN(C(=O)COC2CCC(F)(F)CC2)CC1CNC(C1CC(C#N)C1)=O C1(C(C)O)CCCN(C(=O)CC2CN(C(C3(CO)CCC3)=O)CCO2)C1 c1(C(=O)NC2C(NC(c3cnc(C)[nH]3)=O)CCC2)cc2occ(Br)c2[nH]1 c1(C(=O)NCC(C)NC(C(c2c(C)cncc2)C)=O)cc(Cl)cc2ccncc12 c1(CCCOC(=O)NC(C(=O)NCC)C)ccccc1C N1(C(c2cc(C)oc2)=O)CCC2(CCC2)C(NC(c2cnc3scc(C)n23)=O)C1 c1(CC)cc(NC(=O)NCC(C)CC2CC2)c(C)cc1F CCC(CCCC(=O)NCC(C)(C)C(C)O)NC(c1nccnc1C)=O c1(C(=O)NC(C(CO)NC(CC=C(C)C)=O)C)cnc(O)c2cncn12 C1(C(=O)NCC(C(=O)OCC)C)CN(C(=O)Cc2ccsc2C)CC1(F)F C12(NC(c3ccc(C(C)C)cn3)=O)COC(C1)C(NC(=O)CC1CC1C1CC1)C2 C1(CNC(C(COC)(F)F)=O)CCN(C(=O)C(=O)NC2CC2)CC1(F)F c1(CN(CCOC)CCNC(C2CC23CCOC3)=O)cnc2ccccn12 C1(CCCC(C)(C)C)C(=O)N1.N1(CCN(C2(CCCC)CC2)C)CCOCC1 C1(N2CCCC(C(N(C)Cc3nccn3C)=O)C2)CCCCC1S(C)(=O)=O CC(C)C(C1CCC1)SC(C)C(=O)NCCOCCOC(C)C CC1(O)CCCC1n1cc(CN2CCC2Cn2cc(C(O)C3CC3)nn2)nn1 Cc1cc(C)c(NC(=O)CCCN(C)C(c2nnc(S)n2C)=O)cc1C N1(C(C(CCCCC)O)=O)CCOC2(CCCN(C(=O)Cn3cncc3C)C2)C1 c1(C(=O)NCC2(F)CC(CNC(CC(C)SC)=O)C2)cc2ncccn2n1 N1(C(COCCCC#C)=O)CCC2(COC(CNC(=O)C3=CCOCC3)C2)C1 C(=O)(C(C)=NOCC#N)N(C1(CC(=O)N(C(C#C)C)C)CC1)C C1(C(=O)NC(c2scc(C)n2)C)C=CCN(C(c2ccnc(CO)c2)=O)C1 C(C)(CN=c1[nH]cnc2[nH]ccc12)NC(C(CC)CC(F)(F)F)=O N1(C(CSCC(N)=O)=O)CCC(C2CC2)C1C(=O)NC1CCC(O)C1 C(=O)(CCCC(F)(F)F)NC1CCC(C(=O)NCc2cnc(C(C)C)[nH]2)C1 C(CCCC(=O)N(CC(=O)N(CC(O)C1CCC1)C)CC(C)C)(OC)OC CC1CCc2c(sc3nc(SCc4ccc(N)cc4Br)nc(O)c23)C1 C(N=c1nc2[nH][nH]cc-2c(O)n1)C1CCCN(C(C2CN(C)CC(C)O2)=O)C1 c1(C(N2CC(C(=O)OC)C2)=O)ccc(CNC(C(C=C)O)=O)cc1S(C)(=O)=O N1(C(c2c(CC)onc2)=O)CCN(C(C2CC2CCOC)=O)CC1C1CCC1 N1(C(C2C(CN(C)C)C2)=O)CCCC1(C)CNC(=O)CCCC1(C)N=N1 CN1CC2(CCN(C(C3CN(C(c4ccc(Cl)cc4)=O)C3)=O)CC2)C1 c1(C2C(NCc3cn(CC(N)=O)nn3)C2)cccc(Cl)c1Cl C(CC1CC1)(CC(=O)N(C(C)C)Cc1ccon1)NC(CSCC#C)=O C1(NC(CC(C)SC)=O)CCCC12CCN(C(=O)CCCOC(C)C)CC2 N1(C(C(CNC(C(C(CC)CC)F)=O)(C)C)=O)CCCC2OCCC2C1 C1(C(=O)NC)(NC(c2ccc(C)cc2)c2n(CC)nnn2)CCCCC1 CC(C(=O)NC1COCCN(C(c2ccc(CO)s2)=O)C1)S(C)(=O)=O N1(C(CCNCCCC)=O)CCC(C2(NC(=O)C(C)OC3CCCC3)CC2)C1 c1(C(C)NC(c2cc(CNC(=O)CCc3ccc[nH]3)[nH]n2)=O)ccc(O)nc1 Cc1cc(O)ccc1CNc1ncc(-c2ccnn2C(C)C)cc1O C1(C(=O)NC2(CC=C)CCN(C(c3cocc3C)=O)C2)Cc2nncn2C1 N(C(=NCCF)N1CCCC2(CCSC2)C1)C1CCS(=O)(=O)C1 Cc1ccccc1C(C)C(N1CCCC1C(=O)NCCc1cccc(O)n1)=O N1(C(CCSC)=O)CCOCC2(CC(CNC(C3CCCCO3)=O)CO2)C1 C1(C(N2CCCC(CC(C)C)C2)=O)CN(C(=O)CC(C)F)CC1(F)F N1(C(=O)NCCC(CN=[N+]=[N-])F)CCC2(CC1)OCCc1ccccc12 c1(C(=O)NCCC(C)NC(c2ccn(-c3ccoc3)n2)=O)ccc(C(N)=O)s1 c1(C(=O)OC)cccc2c1CN(C(C)Cc1ncc3ccccn13)C2 N1(C(C2CC(=C)C2)=O)CCc2nc(CNC(c3cccn(C)c3=O)=O)sc2C1 N1(C(CSCCC)=O)CCC(NC(=O)COc2cccc(C(C)C)c2)C1(C)C c1(C(=O)NC2C3CCN(C(CCCNC(N)=O)=O)CC32)c(F)ccc(F)c1F CC1CC(NC(=O)C=CCC2(NC(=O)CC3CC(C)(C)CO3)CCC2)CCS1 C(=O)(CCC(F)F)NCC1(C)CC(NC(C2C(OC)(OC)CC2)=O)C1 N1(C(CC2CCC(=O)N2)=O)CC2(CNC(C3(C4CC4)CCCO3)=O)CCC1CC2 CCC(C)C(C)C(=O)N1CC(F)CC1C1(NC(=O)CC=Cc2cccc(F)c2)CC1 CCC(CCC(=O)N1CCC(NC(c2oc(CO)cc2C)=O)C(F)C1)OC c1(C(C(=O)NC(CCNC(c2c(CC)n(C)cc2)=O)C)C)c[nH]c2ccccc12 c1(C(=O)NC2CCN(C(c3cc(CC)[nH]n3)=O)CC2F)ccc([N+](=O)[O-])c(C)c1 c1(CN(C(C(=O)NCCOC)C(C)C2CCOC2)C)ccc(C(C)(C)C)cc1 N1(C(CCCN(C(C)C)C)=O)CCC(C)C(N(C(=O)Cc2cnsc2)C)C1 C#Cc1cnc(C(N2CC(CNC(C34CCOC(C)(C3)C4)=O)C3CC23)=O)c(C)c1 c1(CNC(NCC(C)NC)=NC)cc(Cl)ccc1OCC(F)(F)F C12(CNC(c3c(CC)nc[nH]3)=O)CC1CN(C(c1[nH]ccc1C1CC1)=O)C2 N1(C(c2c(C)c[nH]n2)=O)CCCC(O)(CNC(=O)CCOC2CC2)C1 c1(C(=O)NCCC2CC(Nc3ncncc3I)C2)cc(F)c(F)cc1Cl CC1(C)CCN(C(c2cc3sccc3[nH]2)=O)C1CNC(C1CNC(=O)N1)=O CC(CN(C)C(C1CCCC1(C)C)=O)N=c1[nH]ccn2nnnc12 C1(C(=O)Nc2ccc(C(=O)NC)cc2)CC2(CC2)CN1Cc1cccc(=O)n1C c1(C(=O)NC(C(C)NC(c2cn(CCC)nn2)=O)C)cnc2ncnn2c1CC CC1Cc2cccc(C(N3CCC(NC(=O)C4=CCOC4)C(O)C3)=O)c2O1 c1(OC)ccc(C)nc1C(N1CCCC1CCNC(C1CCCOC1C)=O)=O C1(C)(NC(C(CC)N(C)C(c2ccccc2C#N)=O)=O)C(C)(C)C1(C)C C(C1=CCCN(C(C2CC(=O)NC2(C)C)=O)C1)NC(C(CN(C)C)O)=O c1(C(=O)NCC2CCC(Nc3c(C)cnc(Cl)n3)C2)cc2ncccc2s1 C1(CNC(=O)Cc2ccns2)CC(NC(c2cc(F)cc(F)c2)=O)C12CCC2 c1(-c2cn(CC(=O)NC(C3CCCC3)CC3CSCCS3)nn2)ccc(Cl)nc1 N1(C(C(CC)=CC)=O)CCN(C(=O)Cc2ccc(O)cc2)CC1CC c1(CC(C(=O)OCC)N(C(C(=O)NC(C)C)c2cncs2)C)cc(Cl)ccc1Cl c1(CC(=O)NCC2(O)CN(C(CN(CC(C)(C)C)C)=O)C2)cccc(F)c1 Cc1cnc(F)c(C(C)NS(=O)(=O)CC2CCN2)c1 C1(C(=O)NC(C)CN(C(=O)C(O)c2ccsc2)C)CCOC1C c1(CNC(C(C)CO)=O)cnn(C)c1C(=O)NCC1COCC(C)O1 N1(C(c2c(CC)[nH]cc2)=O)CCC2CCN(C(c3cnc(CO)nc3C)=O)C2C1 C(=O)(CC(C)(F)F)NC(C)CCN(C(=O)CCc1ccn(C)n1)C c1(OC)cc(C#N)ccc1S(=O)(=O)Nc1ccc(-c2cnn(C)c2)s1 C1(NC(CCNC(=O)C=CCl)=O)CCN(C(c2cccc(N3CCC3)c2)=O)C1C C1(NC(C(C(CC)(F)F)(C)C)=O)CS(=O)(=O)CC1N=c1cc(C)nc(Cl)[nH]1 N1(C(c2nn(C)c(C(F)(F)F)c2)=O)CCC2CCC(NC(=O)CCN3CCC3)C1C2 c1(CNC(C2C(NC(c3ccn(C4CC4(F)F)n3)=O)C2)=O)c(F)cccc1Cl CCCC(C(=O)N1CCC(NC(=O)C(C2CCS(=O)(=O)CC2)O)CC1)S(N)(=O)=O c1(NC(C2N(C(c3cc(CC)ncc3)=O)CC2)=O)ccc2[nH]nc(Cl)c2c1 CC1N(C(c2c(CNC(C3(C)C=CCCC3)=O)cnn2C)=O)CCCC1(C)C C1(C(=O)NCC2C(CNC(C3CC(CC)C3)=O)C2(C)C)(CO)CCCO1 C1(NC2(C(=O)OC)CC2)CC2(C1)CC2C(=O)NC N12CCCC(C1)C(=O)NCC(CC)NC(=O)C2=O.C1(N(C)C)(CO)CCCC1.CCO C1(C(=O)NCCCn2ccnn2)C=CCN1C(c1nocc1Cl)=O C1(C(N2CC(CNC(C=Cc3c(C)n[nH]c3)=O)C(C)C2)=O)CC(=O)NC(C)C1 CC1CN(C(=O)CCn2cnnn2)CCC1NC(c1cc(Cl)cnc1O)=O C=C(Cl)C(C)(C)C(=O)NCC1CCCN(C(=O)C(F)CC2CCCCC2)CC1 Cc1nc2[nH]c(C(=O)NC(C)(CNC(=O)C=Cc3cccnc3)C3CC3)cc2s1 Cc1cc(C(=O)NCC2(C)CCN(C(=O)CN3CCC3C)C2)nc(O)n1 c1(CN2C(CC(=O)NS(=O)(=O)CC3CC3)COCC2)c(Br)cc(F)c(F)c1F C(=O)(C#CC1CCOCC1)N(CC(C)OC(C)=O)C.N12CC(C1)C2=O c1(C(C(=O)NCC2(NC(c3c(CC)n[nH]c3)=O)CCOC2)(C)C)c(C)noc1C C#CCC(CC#C)C(=O)NC1(CO)CN(C(c2nc(Cl)ccc2F)=O)C1 c1(C(=O)NC2CN(C(C=CC(CC)C)=O)C(CC)(CC)C2)cccn2cnnc12 c1(NC(C(c2c(C)scc2)NC(c2csc(CO)n2)=O)=O)ccccc1[N+](=O)[O-] C1(NC(C2CC2F)=O)(CF)CCN(C(c2ncccc2Cl)=O)C1 CC1C(NC(=O)C=Cc2ccc(F)cc2)C(C)CCN1C(C1CC2CCC1O2)=O Cc1cc(O)cc(=O)n1CC(=O)NCC1CCN(C(c2cc3occc3[nH]2)=O)C1 C(=O)(C1=CCCSC1)NCCCN(C(C(CC)OC)=O)CC N1(C(COC2(C)CCC2)=O)CCC(c2cccc(F)c2)C(NC(C2CC2C#N)=O)C1 N1(c2c(C(=O)OC)cnc(Cl)n2)CC2CCC1C(NC(=O)CC1CCC(C)C1)C2 c1(NC(c2cc(C)c(Br)cc2)=O)ccc2c(c1)CCN(C(=O)C(C)(C)F)C2 C1(C)(CNC(c2c(CC)nn[nH]2)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1 c1(C(N2C(CNC(C3CC(OC)(OC)C3)=O)CC(OC)C2)=O)cc(C)cc(C)n1 N1(C(c2cc(OC)c(C)cc2)=O)CC2(CCC(CNC(C3(CCF)CC3)=O)O2)C1 C1(CNC(c2cnc(O)c(F)c2)=O)CCCCN(C(C2C=CCC2)=O)C1 c1(C(C(=O)NC(CC)CN(C(=O)C(C)(C)OC)C)C)c(C)n[nH]c1C C(=O)(C#CC1CCOC1)N1CC(C(C)NC(=O)CCOC2CCCC2)C1 c1(OC)cc(C)cnc1C(=O)NCCCN(C)C(C1CCO1)=O c1(C(N2CCC(C(=O)OC)CC2)=O)c(F)ccc(C)c1Cl.C1(C(C)C)C(=O)O1 N1(C(COC(CC)C)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1CO C1(NC(CCCC#C)=O)CCC(C)(C)CC1CNC(=O)C(CO)N(C)C c1(C(=O)NCC=CCNC(CCCCC)=O)ccc2c(O)nc(=O)n(C)c2n1 CC(C)C(C#N)C(=O)N1CC(NC(c2ccc(-c3ccccc3)cc2)=O)CC1C c1(C(N(CCC(C)NC(c2csc(-c3nc[nH]n3)n2)=O)C)=O)c[nH]c(=N)s1 c1(OCC)ccc(C(=O)NCC(C)(C)CCNC(=O)CC2CCC(=O)N2)cc1Cl C1(NC(c2cc(CNC(c3c(C)cco3)=O)oc2)=O)CN2CCC1CC2 C1(CC(=O)N(CC(F)Cl)C)CC(C)(C)CN1C(=O)CCc1ccn(C)c1 Cc1cccn2ncc(C(=O)NCC3CC(NC(C4(C)CC4(F)Cl)=O)C3)c12 c1(C(N(CCNC(c2ccc(Cl)cn2)=O)C2CC2)=O)cccc(-c2ccsc2)c1 Cc1cc(F)ccc1NC(=O)CNC(=O)CNC(C1(CO)CCCC1)=O N1(C(=O)CC=Cc2ccccc2)CCC(C2CC2)C1CNC(C12CC(CO1)C2)=O C(C)(CC(=O)NC1CC2CC1N(C(c1cnc(N)cn1)=O)C2)(C(F)F)N(C)C c1(OC)n[nH]c(C(=O)NC(C2CCCCN2C(=O)CC2CN(C)C2)C)c1Cl c1(C(=O)NC(c2nc(C3CC3)no2)C(=O)OC)c(Cl)ccc(Br)c1Cl c1(CC=C)cccc(C(N2CCCC(CNC(c3cc(OC)cnn3)=O)C2)=O)c1 N1(C(C)=O)CC(C(=O)NN2CCCC2)C1.C1(C)C=CC(=O)N1C C12(NC(=O)Cc3cncc(O)c3)CCCC1CN(C(=O)C=CSc1nc[nH]n1)C2 c1(N2CC3C(COC)(C3)C2)nc(N2CC=C(C(C)(C)C)CC2)c2c(n1)CCC2 C1(C(=O)Nc2ccc(OC)nc2)CC12CCN(C(=O)NCc1n[nH]c(C)n1)CC2 O=C(CCCCCNC(C1CCOCC1)=O)NCCn1ncnn1 C=CCCCCCCCCCC(=O)N(C)CC1CCN(C(C2CCCN2C)=O)C1 C1(C#CC(=O)N2CC(F)CC2C(N2CC(O)C(O)C2)=O)(CC)COC1 N1(C(c2c(OC)cccn2)=O)CCC(F)C(NC(=O)C(C)C(C)(F)F)C1 C1(C(=O)OC)CCCC1CNC(C1(NC(=O)CC=C)CC1)=O Cc1ccc(C(=O)N(C2CCC(NC(C3COC3)=O)CC2)C)c(C2CC2)c1 CC(O)C(C(=O)NCc1nn[nH]n1)NC(=O)C=CCF Cc1c(NC(C)C)cccc1C(=O)NCC1C2CC2CN1C(=O)CC1CCSCC1 C12(C(=O)NCC3N(C(C(C=C)O)=O)C4C(C3)CCC4)CC3CC(C1)CC(C)(C3)C2 c1(NC(C)=O)cc(Br)ccc1CN=c1[nH]c(COc2ccccc2)cs1 C=C1CCC(C(N2CC3C(CNC(C4(NC(C)=O)CCCC4)=O)C3C2)=O)CC1 N1(C(COC)C)CCN(C(=O)CCN(CCO)CCO)CC1.c12sccc1C(=O)N2 N1(C(c2n(C)nc(Cl)c2)=O)CCC2(C(=O)NC(C3CCC3)C3CCC3)CCCC12 CCCCC(O)C(C)C(=O)N1CC(C(O)C(=O)N(C)CC2CCSC2)C1 c1(C(=O)NCCCCCNC(C2(CCOC)CCC2)=O)cccc(C(C)C)c1 N1(C(c2cc(OCC)no2)=O)CC2CC(C1)C2NC(C1(C)CC1F)=O C1(C(=O)NCC2(C)N(C(COCCCCC)=O)CCC2)Cc2ccc(C)cc2S1 C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CC2=C(CN(C(CCCC(CC)C)=O)C2)C1 C1(CC#C)(NC(=O)C(CCSC)NC(=O)C(C)C2CC2)CCOCC1 Cc1cn2nc(C(=O)N(C)CCN(C)C(C3CC4CCC3CC4)=O)cc2c(=O)[nH]1 C1(C(N2CCC(N(C(C3CCCOC3C)=O)CC)CC2)=O)C2CCC3C(C2)CC13 c1(C(N(CCCCN(C(c2cc(OC)n[nH]2)=O)C)C)=O)ncnc(OC)c1F c1(C(=O)NCCCN(C)C)cc(O)nc2c1CN(C(=O)CCC1CCOC1)CC2 C(=O)(CC(CN(C)C)CC)N1CC(CN(C(C(C2CC2)OCC)=O)C)OCC1 C1(NC(c2occ(C)c2)=O)CC2CCC(C1C)N2C(=O)CCc1cnoc1 Cc1cc(C(N2CCN(C)CC2CNC(c2cnn(C)c2N)=O)=O)nc(O)c1 CC(CCNC(c1cncc(CO)c1)=O)CCNC(C1CCC(=O)N1)=O C12C3CC4C(C3)C14C(=O)N2.C(CCC(=O)N(CC(F)F)C1CC1)C1C(C)C1 Cc1cnc(C(=O)NCC2(O)CCCN(C(=O)CN3CCSCC3)C2)cc1Cl c1(C(N2CCC3(C(NC(=O)CCc4cncs4)C3)C2)=O)cc2c([nH]1)CCCC2 N1(C(C(N)=O)=O)CCC(C(F)C(=O)NC(CO)CCF)C1 N1(C(C(=O)NCC(=C)C)CC2CCCC2)CCOCC1CC1CC1 CCC(CC)C(F)C(=O)N(CC(N1CC(O)(CC(C)C)C1)=O)C(C)C N1(C(C2C(OC(C)=O)C2)=O)CCCC1C(C)(C)NC(=O)C(c1cccnc1)O C1(CCNC(C(CN(C)C)N(C)C)=O)CSCCN1c1ncncc1Br C(=O)(C1CCC(=O)c2cccn21)N1CC(O)(CCNC(c2cncnc2)=O)C1 c1(C(=O)NCC(=O)NCC(CC)CO)ccc(O)nn1 CC1(C)CC(CNC(c2cc(CO)on2)=O)CN(C(=O)CCSC2CCCC2)C1 C#CCCCC(=O)NCC1CCC(C(=O)NC(C2CCOCC2)C)O1 C1(C)(C(=O)NC(C2CCN(C(C3(C)CC(F)C3)=O)CC2)C)COC(=O)OC1 C1(C(N2C(CC(=O)N(C)Cc3ccn(CC)n3)CCC2)=O)CCCN1C=O c1(C(=O)NC2C(CNC(Cc3c(C)n[nH]c3C)=O)C2)cccc([N+](=O)[O-])c1 c1(C(N(C2CCN(C(c3cc(C)nc(O)n3)=O)C2)C)=O)ccc2ncc(C)n2c1 CC(C)CC(O)C(=O)NC1CN(Cc2ccc(C(C)C)nc2)CC1F C1(CC)C(NC(C2COCC(C)(C)O2)=O)CCCN1C(=O)CC(C)C(C)C N1(C(c2cscn2)=O)CCCC2(CCN(Cc3cc([N+](=O)[O-])ccc3O)C2)C1 N1(C(Cc2ccc(OC)cc2C)=O)CCC2(C1)CN(C(=O)C(C)O)CC(C)O2 C1(CNC(C2(CC)CC2(F)F)=O)CCCN(C(=O)CCC2(C)CC2)CC1 c1(C(=O)NC)nc(=NC2CCCC2C(=O)OC)cc[nH]1 N1(C(c2ncc(OC(C)C)nc2)=O)CCOC2(CCN(C(=O)C(C)(C)C)CC2)C1 c1(OC)cc(N)c(F)cc1C(N1CCC(N(C)C(c2csc(C(C)=O)c2)=O)C1)=O n1(CCOC)ncc(C(N2CCOC(CCNC(=O)C(C)=C3CC3)C2)=O)c1C CCC(CC)C(=O)NC1CCCC1CNC(C1(C)CC1(Cl)Cl)=O C(C(=O)NCC1CC(NC(C2CC3CC2C3)=O)C1)(C(F)(F)F)OC(C)=O C1(CCC)(NC(C2CC(Cl)(Cl)C2)=O)CCCN(C(C2CC3CCC3C2)=O)C1 C1(CC(=O)NC2(CNC(c3ncn(C)n3)=O)CCOC2)CCCC2(CC2)C1 Cc1ccc(C(=O)NC2CC2CNC(=O)C(C)(C)c2ccccc2)cc1C(=O)O C(=O)(C1=CCCCC1)NC(CCOC)CNC(=O)CCc1cncnc1O N1(C(CSCCC)=O)CCC(O)C(N(C(=O)COC(C)(C)C)C)C1 C(=O)(CC(C)CC(C)C)NC1CCC(NC(Cc2cc(C(C)C)no2)=O)CC1 CC1CN(C)CC(C(N2CC(CNC(c3cc(Cl)ncc3N)=O)C2)=O)O1 c1(Cc2cccc(NC(CNC(C(COC)OC)=O)=O)c2)ccc(F)c(F)c1 C1(CNC(CCOCCC)=O)C=CCN1C(C1CCCN1C1CCCCC1)=O C(=O)(C(C)S(N)(=O)=O)NCCN(C(C=C(C)Cl)=O)C(C)C C(=O)(C1=CCSC1)N(c1nnc(O)n1C)C(C)C(=O)NCCCC1CCOC1=O C(=O)(C(O)CCNC(=O)Cc1cccnc1)NC(C=C)(C)CC c1(OC)ccc(O)cc1C(=O)NC1CC(F)(CNC(C2CCOC2(C)C)=O)C1 c1(OC)cc(OC)nc(C(=O)NC2(CNC(C3CCCC(C)C3)=O)CCCC2)n1 C(=O)(C1=NN(CC=C(C)C)C(=O)CC1)NC(CC)CNC(=O)C(C)=CC(C)(C)C C1(NC(c2cn(CCO)nn2)=O)CCOC1C(=O)NC1CC(Cl)(Cl)C1 N1(C(C2ON=C(C)C2C)=O)CC2CN(C(c3conc3C)=O)CCC12 C(=O)(C(C)(C)C(C)C)N(CC(CN(C(c1c(CC)[nH]cc1)=O)C)O)C c1(CC)ccc(C(C)=CC(=O)NCC2(C(N)=O)CN(C(C3CC34CC4)=O)C2)cc1 N1(C(c2c(C)scn2)=O)CCC2CC(NC(C3CC4CCC3C4)=O)CCC2C1 C(=O)(C1=CS(=O)(=O)CCC1)NCCC(C(C)C)NC(c1cc(OC)nc(Cl)c1)=O N1(C(c2ccc(COC)cc2)=O)CCCC(O)(CNC(=O)Cc2ccsc2C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CC(NC(C=Cc2c(C)coc2C)=O)C1 Cc1nn(C)c(C)c1C(N1CCCC1(C)C1CCN(C(=O)C(O)C2CCC2)C1)=O Cc1cc(F)ccc1CC(N1CC(N(C(=O)CC2CCC(C#N)C2)C)C1)=O CCC(C)CC(C)NC(=O)C(O)C1CN(C(C2CCC(=O)O2)=O)C1 C12(NC(c3cc(SC)c(C)o3)=O)CCN(C(c3cnco3)=O)CCC1C2 C1(NC(c2cnc(C)nc2)=O)CCN(C(c2cnn(C)c2)=O)CC12CCC2 C1(NC(C=CC(=O)OCC)=O)CCC12CN(C(C1(C)C=CCC1)=O)C2 Cc1c(C(=O)N(C(CNC(=O)CCN(C)C2CC2)C2CC2)C)sc2nccn12 CCCC(O)C(=O)N(C(CNC(C1(C)CC1Br)=O)C1CC1)C C(=O)(C(C)(C)CCOC)NCC(CC=C)NC(c1cc(CC2CC2)on1)=O C1(NC(=O)C2=CCCC2)(CO)CCN(C(=O)CCOc2ccc(F)c(Cl)c2)CC1 c1(CC2CC(NC(C)=O)CN2C(c2csc(C(N)=O)n2)=O)cccc(F)c1C#N C1(C(=O)NCCC(C)NC(c2cc(CC(C)C)[nH]n2)=O)CC2CCC(C1)C2O CCCCC(C)C(=O)NCCC(C)CCNC(C1(OC)CCCCC1)=O c1(C(N2C(CCNC(CCOC)=O)CCC2)=O)cnc2c(c1)CCS(=O)(=O)C2 c1(NCC(C)(C2CC2)NC(=O)CC2CCCCC2O)ccc([N+](=O)[O-])c(C#N)c1 c1(C(N(C(C)CNC(=O)CC(c2cccc(F)c2)C)C)=O)cc2n(n1)CCCN2 C12(CNC(C(C)SCC)=O)CC(NC(=O)COCC(F)(F)F)(CO1)C2 c1(C(=O)NCC=CCC(=O)N(CC)Cc2nncs2)cc(C2CC2)on1 N1(C(C2(SC)CN(C(CCC(CC)=O)=O)C2)=O)CCCC2(C=CCO2)C1 C1(CNC(CC2CN(C)C2)=O)CCCN(C(c2cncc(N)c2)=O)CC1 Cc1ccc(OCC(=O)NCC2C=CC(NC(C3(C)COC3)=O)C2)c(C)c1 C=CCCC(C)(C)C(=O)N1CC2=C(C1)CN(C(=O)Cn1nc(Cl)ccc1=O)C2 c1(C(=O)NC(C2CCN(C(C3C(C#C)C3)=O)C2)(C)C)cccc2nn[nH]c12 Cc1ccc(O)cc1C(N1CC(C)(C(=O)NOCCF)C1)=O c1(C(=O)NCC2N(C(c3ccc(SC)o3)=O)CC=C2)nnn2c1CSCC2 C1(CN(C(c2c(C)scn2)=O)C)CCCC(NC(c2ccn(C3CC3)c2C)=O)C1 C(=O)(C(CCC1CCCC1)N(Cc1scnc1C)CC1CC1)NC(CC)C N1(C(c2c(COC)cccc2)=O)CC2CCN(C(c3coc(Cl)n3)=O)C(C2)C1 c1(C(=O)NCC2CCN(C(=O)COC3CC3)C2)c[nH]c2ccncc12 N1(C(c2cc(COC)sc2)=O)CC2(CC2)CC1CNC(=O)C(C)C(F)(F)F CC(C)C(CCNC(C1CC1(Cl)Cl)=O)NC(C1(CC(C)=O)CCCC1)=O Cc1cc(N)ccc1C(N1CC=C(CNC(c2ccnc(C3CC3)c2)=O)CC1)=O C#Cc1ccc(C(=O)NC23CCC(C2)N(C(C2(OC)CCC2)=O)C3)cc1F Cc1c(C(N2CCC(N(CCO)C(c3cccnc3)=O)C2)=O)[nH]c2ccccc12 Cc1cc(CCC(=O)NCC2(F)CC(NC(C3CC4(CC4)C3)=O)C2)cc(C)c1 C1(CCC(=O)NCCC(=C)CNC(c2cnc(Cl)c(Cl)c2)=O)CCCC(=O)N1 CC(C)CCCCCC(=O)NC1C=CCN(C(c2ccc(CN(C)C)c(F)c2)=O)C1 C1(CNC(C2C(C)CCO2)=O)CN(C(=O)CCCCN(C)C)CC(C)(C)O1 C#Cc1cccc(C(N2CC3CC(C2)N3C(=O)C(C2CCC(=O)N2)C)=O)c1F O=C(C1=CNC2=NCCC2=C1)NC1CN(C(C2CCCC3(CCC3)O2)=O)C1 C=C1CCN(C(=O)C=Cc2cn(C)nn2)C(C(=O)NCCOC2CCC2)C1 NC1(CNC(c2oc(-c3ccccc3)nc2C#N)=O)CC2CCCC12 N1(C(=O)OC(C)(C)C)CCOC2CC(CC3CCCCO3)CC12 C(C1=NOC2COCC12)NC(C(CC(F)F)N(C)C(C1CC2CCC1CC2)=O)=O N1(C(C2(CCN(C)C)CC2)=O)CCN(C(C2CCS2(=O)=O)=O)C(CF)C1 c1(C(=O)O)ccc(Br)c(CN(CCCCC2N=N2)C2CC2)c1 c1(C(N2CCCC(CNC(CCC=CC)=O)CC2)=O)ccc2c(c1)C(=O)CCS2 CC1CC2(CCN(C(=O)C(C)(F)C(C)(C)F)CC2)CN1C(=O)CCCCN(C)C C1(NC(C(C2CN(C(=O)C3=COCC3)C2)OC)=O)(CO)CC2CCCC12 C(=O)(C(C)CC(=O)OC)N1CC(NC(c2cnn(CC)n2)=O)(CF)C1 C=Cn1nncc1C(=O)NC1CCCCC1CNC(=O)COC N1(C(C(COCC)C)=O)CCC(F)(F)C(CNC(=O)C=CCO)C1 CC1SCCCC1C(N1CCCCC1C(=O)NCCCCN(C)C)=O CCC(C(=O)NCCCCCN(C(=O)COCC1CCCC1)C)n1nccc1C C(CCC(=O)NCC(C)(CO)n1cc(Cn2cc(Cl)cn2)nn1)NC(C)=O c1(C(N2C(C)CCC(CNC(CCC(=O)OC)=O)C2)=O)cnc(O)n(C)c1=O C1(C(=O)NC2CCC(NC(C3(C(F)F)CC3)=O)CC2)CC2(C1)CC2(F)F C=CC(C)CC(=O)NC1C=CCCC1C(=O)NCc1ccsc1 C1(CNC(C(C)(C)NC(=O)CCCn2cc(CO)nn2)=O)CC12CC2(F)F c1(C(=O)NCC(C(=O)N(CCSC)CC)C)cnc(O)n1CC CN1CC(C(=O)N(CC(=O)Nc2cncc(F)c2)CC2CC(C#N)C2)NC1=O c1(OC)c[nH]c(C(=O)N(C(C)CNC(c2c[nH]cc(Br)c2=N)=O)C)cc1=O c1(NC(C)=O)cccc(NC(=O)NCc2coc(Cc3ccccc3)c2)c1 c1(N2CC3CC(NC(C4CCCC(C)(C)O4)=O)C3C2)cnc(C#N)c(C#N)n1 Cc1ccc(OCC(=O)N(CC(C)NC(=O)Cc2cc(Cl)cnc2C)C)c(C)c1 c1(C(N(CCC(C)NC(C2CCNC2=O)=O)C)=O)cccc(C2CC2)c1Cl c1(C(N2C(CNC(c3[nH]ccc(=N)n3)=O)CC2)=O)cc(Cl)cc(F)c1F N1(C(C=CC=CC)=O)CC2CCC1CN2C(=O)CN1CSCC1=O c1(CCCCC)cccc(CCc2nc(-c3coc(SC)c3)n(CCF)n2)c1 C(=O)(CC(C)(C)C(C)(F)F)N1CC(O)(C(C)NC(C2CC2C#N)=O)C1 N(C1CCOc2cc(F)ccc21)C(C1CCCN1C(c1cc(=O)cco1)=O)=O C(=O)(C(CC(F)(F)F)c1ccco1)NCC(=O)N(C1(c2nn[nH]n2)CC1)C C1(C(=O)NCc2ncc(C#N)o2)CCN(C(=O)CC2CC(F)C2)CCO1 N1(C(C2CC(C#N)(OC)C2)=O)CC2CC(NC(C3CC(OC)C3)=O)C2C1 c1(OC)cc(N)c(C(=O)NC2CC(NC(c3cscn3)=O)C23CCC3)cc1OC C(=O)(C1=CCCCCC1)NCC1C(C)CCN(C(C2C(C)(C)C2(C)C)=O)C1 CN1CC(NC(=O)C(CNC(c2cc(C3CC3)on2)=O)CC2CC2)CC1(C)C c1(C(N2CCCC(CCNC(C=CCCC)=O)CC2)=O)ccnc(S(N)(=O)=O)c1 c1(CCC(=O)N(CC(CC)OC)CCNC(=O)C=CC2CC2)csc(=N)[nH]1 c1(C(C(=O)OC)NCC2C(C)C2C)ccccc1Br c1(CC)[nH]nc(Cl)c1C(=O)NC1CC(C)(NC(C2COC(C)(C)C2)=O)C1 C(C(O)CC(C)(C)C)NC(C(CNC(CSC)=O)CC1CC1)=O c1(OC)cccc2[nH]c(C(=O)NC3CCC(C)N(C(=O)CC(C)(F)F)C3)cc12 N1(C(C(C)CS(C)(=O)=O)=O)CCC2CCN(C(c3ccnn3CCF)=O)CC2C1 C12(C(=O)OC)COC(CF)(C1)C2.S1(=O)(=O)CC2(CCC2)N1 O(NC(=O)C(CC1CC1)NC(C1CC1C(C)(C)C)=O)CCCOC CC(C)CC(CNC(C1CC(N2CCOCC2)C1)=O)NC(C1(C)C=CCC1)=O CC1CCc2nc(N(C)CCc3cnccn3)[nH]c(=NCCCN(C)OC)c2C1 c1(-c2cccc(NCc3cc(C(F)(F)F)[nH]n3)n2)cccc2c[nH]nc12 c1(C(=O)NC(C)C(C)NC(=O)CCCCN2CCCCC2)cc2sccc2s1 c1(C(=O)NC2(C3CCN(C(CC(C)n4ccnc4)=O)C3)CC2)csc(C#N)c1 C#CCCCCC(=O)NCc1cnn(C)c1C(=O)N(CC(C)CCC)C N1(CCNC(C2CC(F)(F)C2)=O)CCN(C(C2CC3CC2C3)=O)CC1 C1(C(=O)NC(C2CN(C(c3ccc(CO)o3)=O)CCO2)C)(CO)CCCCC1 CN1CCCC1CCC(N1CCC(CC(=O)NCCC(N)=O)C1)=O c1(C(N2CC(F)(CC(=O)N(CC)Cc3ccccc3)C2)=O)ccc2nncn2c1 C1(O)(CN(C(C2(OC)CCSC2)=O)C)CCCN(C(=O)CS(=O)(=O)N(C)C)C1 C1(CNC(=O)C(O)c2ccco2)CC2CCC1N(C(c1nc(F)ccc1Cl)=O)C2 N1(C(c2c(CC)[nH]cc2)=O)CCC2CN(C(=O)CCCN3CCCC3)CC2CC1 Cc1nc(O)ccc1C(=O)NC1CCCN(C(c2ccc(N)c(CO)c2)=O)C1C Cc1ccc(OC(C)C(=O)N(C(C)CN(C(=O)C2=C(Cl)CC2)C)C)c(C)c1 N#CC1(NC(c2cc(Br)cnc2Br)=O)CCN(C(c2cc(F)nc(F)c2)=O)C1 CC1CN(C(=O)CSCc2cccnc2)CCC1N(C(=O)C=CC(F)F)C c1(OC)ncc(Cl)c(=NC2CC(NC(c3ccn(CCN(C)C)n3)=O)C2)[nH]1 C1(CCNC(C(C(C)C)F)=O)CCN(C(C23CCC(CC2)CC3)=O)CC1(F)F C1(NC(C2CC(CCC)C2)=O)CCN(C(c2cnc(SC)nc2)=O)CC1O C1(C(=O)NC(CNC(CCOCC#C)=O)C)Cc2ccccc2C1C C1(NC(CC2CC(C)(C)C2)=O)CN(C(C2CCC(C(F)(F)F)C2)=O)CC1O C12(NC(c3cccc(C(C)=O)c3)=O)CC(C(=O)NCc3cn[nH]c3)(C1)OC2(C)C C(CN=c1nc(N2CCC(C3CC3)C2)c2c([nH]1)CSC2)N1C(=O)OCC1 C(=O)(CCCC(=O)NC(CO)C(C)NC(c1ccc(C(C)C)cn1)=O)NCCC N1(C(CC(=C)C)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC1c1cn[nH]c1 c1(C(N(CCNC(C(C)OCC=C)=O)CC)=O)ccccc1-n1cccn1 Brc1c[nH]nc1C(c1nnnn1CCCC1CC1)NCCCC1CCCCC1 N1(C(c2ccc(C)o2)=O)CCCC2CCN(C(=O)CC3CC(C)(C)C3)CC12 CC1CN(C(c2coc(CO)c2)=O)CC(C)N(C(=O)C(c2ccncc2)C)C1 CCCC(CCC)CC(=O)N1CC(CCNC(c2[nH]cnc2C)=O)OC(C)C1 N1(C(c2nn(CC)c(O)c2)=O)CCC(O)(CCNC(C2CC(Cl)(Cl)C2)=O)CC1 c1(C(N2CC3C(NC(C(C)OCCCCCC)=O)C3C2)=O)cnc(N)c(Cl)c1 c1(N(C(COC)=O)C)nc(N(CCCn2ccc(=O)cc2)C)nc(C)n1 Cc1cc(Br)ccc1CN1CCCC1C(=O)NCCCCCO c1(C(N2C(CNC(CC(CC)SC)=O)CC2)=O)cnc(C)c(C)c1 c1(C(C(F)(F)F)NC(=O)Cc2ccn(C3CCOCC3)n2)ccc(Cl)cc1 C(=O)(CCCCCC1CC1)N1C(C)(C(=O)NCC(F)Br)C=CC1 c1(CC)nn(C)c(Cl)c1C(N1CCC(NC(c2ccccc2)=O)C(CO)C1)=O C(C(C(C)(C)C)NC(C1(C)CCSCC1)=O)NC(c1c(CC)scc1)=O N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CN(C(c3cc(C(F)F)no3)=O)CC12 C(=O)(C(CC(C)C)Oc1nn(C)cc1C#C)NCC(=O)NC(C1CCCC1)C#C CC(C(=O)NC12CCC(C1)N(C(=O)Cc1ccc(F)cn1)C2)C(F)(F)F N1(C(c2snc(C)c2Br)=O)CC2ON=C(CNC(C3(C)CC3)=O)C2C1 C(=O)(C1=CCOCC1)NCCNC(C(C(=O)OC(C)(C)C)OC)=O.C1CCN1 CCC(C)N=c1cc(NCCC2COC(=O)N2)nc(C(F)(F)F)[nH]1 C#Cc1cnn(CC(=O)NCCN(C(c2cccnc2-n2nccn2)=O)CC)c1 N12CCC(C)(C)C1C(=O)OCC2=O.C(CS(C)(=N)=O)N.C1(OC)CCCC1 CC1CCNCCC1N(c1ccc(S(N)(=O)=O)o1)C(c1c(Cl)cccc1Cl)=O N1(C(CC(C)F)=O)CCC2(CCC2NC(c2ccc(C(C)(C)C)c(Cl)c2)=O)CC1 CCCCCCCCCN1CCOC(C)(CNC(=O)CCc2nc(C)no2)C1 N1(C(C(CC)=CCCC)=O)CC(C(c2ccccc2)NC(=O)C(C)(F)F)C(C)(C)C1 C1(NC(C(=O)NCCOC)=O)CC2CCC1(CNC(C1CC(S(C)(=O)=O)C1)=O)C2 C=Cn1nccc1C(=O)NCCCCCNC(=O)Cn1nc(C)oc1=O CC1CNCCC1N(C(=O)C(=O)NCC(C)(C)c1cccs1)C C(C(COC)C(C)C)(c1n(CC)nnn1)NCc1ccc(OC(F)F)c(F)c1 N1(C(c2oc(CC)c(C)c2)=O)CC2CCN(C(c3ccc(Cl)cc3O)=O)C2C1 C1(CNC(C2CCCN(CC)C2)=O)CCN(C(=O)CC2(CO)CC2)CC1C c1(C(=O)NC2CC(N(C(C3(OC)CCCC3)=O)C)C2)nc2nccc(C)n2n1 N12CCOC(C)C1C2.N1(C(C=CC)=O)CCC(C(=O)NC)(OC)C1 C1(CN(C(CSCC#C)=O)CC)CCN(C(C)=O)C1.C(=O)(COCCF)NCC CC(CS(C)(=O)=O)C(=O)N1CC2(CCC2NC(c2ccc(F)cc2F)=O)C1 C1(n2cc(Cn3cccc3)nn2)(C(=O)NCC2(C)CC2(Cl)Cl)CCOCC1 C1(CNC(COC(CC)(C)C)=O)CCCN1C(=O)C(C)(C)c1ccns1 C1(OC)CCC(C(N2CCCC2CN(C(=O)CC(C)(C)C2CC2)C)=O)CC1 N1(C(CCCCC(=O)OC)=O)CC2C3CCC(C2C1)N(C(c1c[nH]nc1C)=O)C3 C(C1=NOC2CCCCC12)n1cc(C2CN(C(=O)CC3OCCO3)C2)nn1 N1(C(=O)CC2=CCCC2)CCC2(CCCCC2NC(=O)C(F)(F)CC2CC2)CC1 C(CCCCCNC(c1sccc1CC#N)=O)N(C)C(C1(C)COCCO1)=O C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CN(c2c(C)cc([N+](=O)[O-])cc2)C(C)CC1 c1(C(N2CC(=C(CNC(c3ccn(CC)n3)=O)F)C2)=O)ccc(O)c(N=[N+]=[N-])c1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC(F)(CNC(C(C)OCCOCC)=O)C1 C1(SC)CN(C(c2cccc(C3CCCOC3)c2)=O)CC1NC(=O)CCF CCC(CC(=O)N1CCC(C)(C)C(C(=O)NCC2=NOC(C)C2)C1)C(F)F N1(c2c(C(N)=O)cnc(Cl)n2)CCCC2(NC(C3CCOC3)=O)CC2C1 C1(C)(CC(=O)N(CCCN(C)C)CC)CCN(C(=O)Cc2coc(C)n2)C1 c1(CCCC(=O)N(C)CCC2CCCN2C)ccc2c(c1)OCO2 c1(OCC)cc(CNC(C2CC(NC)C2)=O)c2c(c1)CC(C)O2 Cc1cc(O)c(C(C)C)cc1C(=O)N(C1CN(C(C2CC=CCO2)=O)C1)C C1(NC(Cn2nnc(C(C)(C)C)n2)=O)CN(C(c2ccoc2)=O)CCC12CCC2 C1(CNC(C2C(C)=CCS2)=O)CCCC2CN(C(c3occc3C)=O)CC12 c1(C(=O)NC(CNC(CC=CC)=O)C)cnc(O)cc1C(F)(F)F c1(NC(c2nc(CC)oc2)=O)ccc(-n2cc(C(N)=O)nn2)cc1 c1(SCC(=O)NCCCN(C(C2(C)C=CCCC2)=O)CC)ccc(OC)cc1 Cn1cc2c(n1)CCN(C(C1CC1NC(c1cccc(I)c1[N+](=O)[O-])=O)=O)C2 C1(C(=O)NCC2(OC)CCN(C(=O)COC(C)C)C2)OCC2CCCCC12 CCCCC(F)(F)C(=O)NCCc1n[nH]cc1C(=O)NC1CC2CC2C1 Cc1cc(C(N2CCN(C(c3cnc(O)s3)=O)CC2CO)=O)c2n[nH]cc2c1 C1(C(N2CCC(COCC)CC2)=O)CN(C(C2(OC)CCSC2)=O)CCN1C C#Cc1ccc(NC(=O)CCCC(C)(C)NC(c2ccnn2C)=O)c(C)c1 c1(OCC(N2CCCC(NC(c3ccn(C)n3)=O)C2)=O)ccc(F)c(F)c1 C1(CNC(CC2(OC)CCC2)=O)CN(C(C2CCOC(C)(C)C2)=O)CCC1(C)C C1(C(C)NC(=O)CCOC2COC2)CCN(C(=O)C(C)N2CCCC2)CC1 c1(CC(=O)NC(C2CCN(C(COC(CC)(C)C)=O)CC2)C)ccc(C#N)cc1 C(=O)(C(C(=O)N(CCN(C(=O)C(O)CC1CC1)C)C)C1CC1)OC.N1(CC)CCCC1 c1(OC)c(F)ccc(F)c1C(=O)Nc1cnc2n1CCOC2 C1(CNC(C(N2CCNC2=O)C)=O)CCCN(C(=O)CN2CCC(O)CC2)CC1 C(=O)(CCC(=O)NC(CC(=O)NC(CN(C)C)CO)C1CC1)NC c1(C(N2C(C)(C(=O)NC(C(C)SC)C)CCC2)=O)cc(C)c(F)cn1 c1(C(=O)Nc2cccc(-c3n(CC)cnn3)c2)sc2cccnc2c1Br CC(C)CC(F)(F)C(=O)NCCC1CCN(C(c2ccc(OCCF)cc2)=O)C1 Cc1cccc(C(N2CC3CC2C3C(=O)Nc2cc(Cl)ccn2)=O)n1 C1(n2cc(-c3nc(CC)sc3)nn2)(C(N2CC(=O)N(C)CC2)=O)CC(C)CC(C)C1 C1(NC(C(=Cc2c(CC)[nH]c(O)n2)C)=O)CC12CCN(C(=O)C(F)C(C)(C)O)CC2 C(=O)(CCCCCCCNC(=O)OC(C)(C)C)N(C(C)C(=O)NC)CC Cc1cc(C(=O)NCCNC(=O)CC2CCCC(C)(C)O2)c2ccccc2n1 CC1(C(N2CCN(C(=O)C(=O)Nc3ccc(F)cc3)CC2)C2CC2)NC(=O)NC1=O C=C=C(C)CC(=O)NCCC1CSCCN1C(=O)CN1CCCCC1 C(C1c2ccccc2CCN1C(C1CC(=O)N(O)C1)=O)NC(c1cscn1)=O C1(NC(C2(CCOC)CCCC2)=O)CCN(C(c2ccncc2)=O)C1C1CC1 C(c1ccncc1)=CC(=O)NCC(C)CN(C(=O)CN(C)C(N)=O)C c1(CNC(c2nnnn2C(C)CC)CCC)ccc(OC(C)COC)cc1 N1(C(c2cc(C)nn2C)=O)CCC2(CCCC2NC(=O)Cc2cccnc2O)C1 n1(C(C)C)cnc2c(NC3CC3C)[nH]c(=NCc3cnccn3)nc12 C1(NC(C(C)=CC)=O)CCC12CN(C(=O)CCc1ccc(F)cc1)C2 C(CN=c1cc(C)nc(C(=O)OC)[nH]1)N(C(CC(CC)C(C)C)=O)CC1CC1 N1(C(c2c(C)nc(C)[nH]2)=O)CC(CNC(C23CCCC2C3(F)F)=O)C(C)(C)C1 C1(NC(c2cncc(SC)c2)=O)CCC(C)N(C(=O)COCCCC(C)C)C1 N1(C(C2(CNC(C3COC(C4CC4)C3)=O)CC(=C)C2)=O)CCCNC(=O)C1 C1(CSC)COCCN1c1nnc(CCCS(N)(=O)=O)n1Cc1ccccc1 c1(Nc2c(OCC)cc(F)cc2)nccc(=NC2CC2c2cncn2C)[nH]1 c1(C(N2CC(NC(CC(C(=O)OC)C)=O)C2)=O)cncc2ccccc12 C1(C(=O)NC2OCCN(CC)C2)CCC2(CC1)CC2.c12cc(ccn1)C(=O)OC2 N1(C(CCC(=O)OC)=O)CCC2(CC1)CC(C(=O)Nc1cccc(O)c1Br)CO2 N#CC1CN(Cc2cncs2)CC1NC(c1cnc(Cl)s1)=O N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C(NC(c2n[nH]c(C)n2)=O)C1 c1(CN(CC)Cc2ccc(-n3cccc3)cc2Cl)nn(C)cc1S(N)(=O)=O NC(=O)CC(C(=O)N1CCC(n2cccn2)C1)NC(c1ccc(C(N)=O)nc1)=O N1(C(c2ccc(C(N)=O)nc2)=O)CC2CC(NC(C3CCSCC3)=O)C1C2 C1(CC(=O)NCC2(O)CN(C(c3cc(CC)n(C)n3)=O)C2)NC(=O)CN(C)C1=O C(C)(CC(=O)N(CCNC(c1ccnn1CCN(C)C)=O)CC1CCCC1)SC Cc1ncc(C(=O)NC(C2CCN(C(c3cc(C4CC4)[nH]n3)=O)C2)C)n1C CC(F)(F)C(C)(C)C(=O)NC12CCCN(C(c3cncc(Cl)n3)=O)CC1C2 c1(C(=O)NC2CCN(C(c3cnc(C(N)=O)s3)=O)CC2F)scc2c1CCCC2 c1(OC)ccc(C(N2CCC(O)(C(C)NC(C3CC(C)(F)C3)=O)CC2)=O)c(F)c1 Cc1n[nH]c(C)c1SCC(=O)N(C)CC1CCCN(C(=O)CC2CC2(C)C)C1 c1(NC(C2(CCNC(CSC)=O)CCCC2)=O)ccc(CNC2CC2)nc1C c1(C(=O)NC23CN(C(c4ccc(C=C)cc4)=O)C(C2)C3)ccc2nc(Cl)nn2c1 N1(CC(=O)NCC(C)NC(c2ccc(COC)o2)=O)CCOCC1=O N1(C(C(CC)=CC)=O)CC2(C1)CN(C(C1CCC3CC13)=O)CCO2 N1(C(C2(OC)CCC(C)C2)=O)CCC2(CC1)CCN(C(=O)CS(=O)(=O)C(C)C)C2 C(CC(C)(C)CNC(C1CCCCO1)=O)NC(C(C)Cc1cnc[nH]1)=O C1(C(NOCC(=C)C)=O)CC(C)CCN1C(=O)C(C)C(=O)OCC S(=O)(=O)(c1ccc(C)cc1Br)NC(C1(CC=C)CCCCCC1)=O S(=O)(=O)(c1ccc2c(c1)CCCN2C(=O)Cn1cc(S(C)(=O)=O)cn1)N(C)C c1(C(=O)NC(CCC)C(=O)N(C(C)CCO)C)ccc2[nH]ccc2n1 C(=O)(C(C)(C)CCCF)NC(C)CCCNC(=O)COc1ccc(F)nc1 C(CCN=C(NCC1CCC(F)(F)C1)NCC1CC1)N(C(C)C)C(=O)NC1CCC1 C=CC1CN(C(c2cn(C)nc2C2CC2)=O)CC1NC(C1(CC)CC1)=O C#CCC(CC(F)F)C(=O)N(C1CN(C(=O)C(C)CC2CCCC2)CC1(C)C)C N1(C(Cc2cc(C)on2)=O)CCC(C)N(C(=O)CCCC(F)F)CC1 N1(Cc2c3ncn(CC(CCC)O)c3ncn2)CC2CCCC(CO)(C1)C2(F)F Cc1cccc2cc(C(=O)NCCOC(C)(C)CNC(=O)Cn3ncnn3)nn12 N1(C(c2ccn(CC)c2C)=O)CCCN(C(=O)C(C)NC(=O)OC(C)(C)C)CC1 c1(OCCNC(Cc2n(C)ccn2)=O)cnc(-c2ccc(F)cc2)cn1 S(=O)(=O)(c1cn(C)c(=O)n(C)c1=O)NC(CCSc1cc(OC)c(Cl)cc1)=O C1(CNC(c2ncc(C(F)(F)F)cn2)=O)CC(O)CCN1S(=O)(=O)C1CC1 C1(C(=O)NC(C)CCCCNC(C2CC2Cl)=O)CCC2CC1C2(C)C CC(C)CC(O)CC(=O)N1CCOCC1CNC(c1scnc1C(F)(F)F)=O c1(C(N2C(C(=O)NC34CC(C(=O)OC)(C3)C4)CCC2)=O)cnc2cc[nH]c2c1 CCCCC(F)(F)CNC(=O)NCCN1CCC(N=[N+]=[N-])CC1 C(=O)(C#CC(=O)N1CC(O)(C(=O)NCC2(N(C)C)CCCC2)C1)N(C)C N1(C(C(C)S(C)(=O)=O)=O)CCC(F)(F)C(CNC(C23CCN(CC2)C3)=O)C1 C1(c2ccc(OC)cc2)C(C(=O)NCC=CC2CCCC2)CC(=O)N1C1CC1 c1(NC(c2cccc(CC)c2)=O)ccc(OSc2cccnc2)c(Br)c1 C12(C(=O)NC3C(NC(C4(C)CCC4)=O)COC3)CCCN(CC1)C2 c1(C(N2C3C(NC(CS(=O)(=O)N(C)C)=O)CC(C3)C2)=O)nn(C)c2c1CCC2 c1(C(=O)NC2CC(NC(CN(C(C)=O)C)=O)C2)c(C)ccc2c1CCCN2 C(CC(C(=O)N1CC([N+](=O)[O-])C1)NC(=O)COc1ccsc1)OCC N#CCC(C(=O)NCC1CC1CNC(C12CC(C(F)F)(C1)C2)=O)c1ccccc1 C1(NC(c2cc(Cl)c(F)cc2O)=O)CN(C(C2CCOCC2)=O)CCC12CCC2 C#CCCCCCCC(=O)NCC(C)N(C(=O)C(C)(C)C(C)(C)O)C c1(C(N(C2CCN(C(c3cc[nH]n3)=O)C2)CC)=O)ccc(S(N)(=O)=O)cc1F C(C(=O)N(CC(C)O)CCOC)(C(C)O)NC(c1c(CC)[nH]cc1)=O C=CCC(CNC(c1cc(F)cnc1O)=O)C(=O)NCc1cnccc1C c1(C(=O)NC(CC)CN(C(c2[nH]nnc2C2CC2)=O)CC)cncc2[nH]ccc12 CC(C(=O)N(C)CCN(C)C(C1CNC(=O)C(C)(C)C1)=O)C(F)(F)C(F)F c1(C2C(C(N3CCCCC3C3CC3)=O)C2)c(Cl)cc(Cl)cc1Cl c1(C(=O)NCCNC(C)=O)cnc2cc(-c3ccc(O)cc3)ccc2c1Cl C(CNC(C1CC(C)N1C(C1CC(=C2CCC2)C1)=O)=O)(C(F)(F)F)OC C(=O)(C(O)CC(C)C)NC(C1CCCC1)CNC(C=Cc1ccc(SC)s1)=O C=CCC(CC(F)(F)F)C(=O)NC(c1cccnc1F)C c1(C(=O)NCC(C)(C)NC(C2C(C(C)C)OCC2)=O)cccc2c1COCC2 Cc1ccncc1CC(=O)NCCCC(C)NC(=O)Cc1ccsn1 C(C(=O)NC(C)C=CC(=O)NC1C=CCCC1CO)(C(C)(C)C)OC N1(C(c2nn(-c3ccc(F)cc3F)c3c2CCC3)=O)CCS(=O)C2(CCC2)C1 C1(C(N2CC(=CC)C2)=O)CCCN(C=O)CC1.c1(OC)ncccc1F N1(C(C2CCN(C(c3nc(C)sc3)=O)C2C)=O)CCCC(C)CC1 c1(C(=O)NCCN(C(c2c(N)cc(Cl)nc2)=O)C2CC2)cncc2c1CCC2 c1(C(C(=O)NCC(C)(O)CNC(C2CC(=C3CC3)C2)=O)(C)O)cccc(F)c1 C1(NC2C(CC=C)C(NC(=O)OC(C)(C)C)C2)CC(O)CN(Cc2ccco2)C1 c1(C2(NC(C3N(C(C4N(CC)CCC4)=O)CCC3)=O)CC2)cc(Cl)cc(Cl)c1 C12(C(=O)NC3(COC)CCC3)CCCC1N(C(=O)CC1COCC(C)O1)CC2 C12CCCN(C1)C2=O.CC(C)C(C)(C)c1cn(CC(=O)Nc2ccc(Br)s2)nn1 C1(NC(C(C)=C2CC2)=O)CN(C(=O)C(C2CCOCC2)C)CC1c1nccn1C Cc1cnn2cc(C(N3CCCC(CNC(C4CCC(=O)N4C)=O)C3)=O)cnc12 Cc1nc(C)c(C(=O)NCC2CN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)s1 C(CC(C(=O)NC1CCCC1)OC)N(CCC(=O)NCC)C.C12CC1(C)CNC2=O c12cnc(nc1)C(=O)NC2.N1(C(C2CC(CCC)C2)=O)CCCCC1CN(C)C N1(C(C(CC)SC)=O)CCC(CCN(C)C(c2ncoc2C(F)(F)F)=O)CC1 C1(NC(CC(C)F)=O)CN(C(=O)COCC2CC2)Cc2ccnn2C1 c1(CC)ncnc(N(C2CCCN(C(C3(CO)COC3)=O)C2)C)c1F C1(C(=O)NCC2(C(=O)OC)CCC2)CCC(NC(=O)COC2CC2)CC1 c1(C(C(=O)N2C(CNC(c3nncs3)=O)CC2)CO)ccc(Cl)cc1 C1(C(=O)NC2C(C)N(C(=O)CC3CC3)CCC2)CCC2(CCC2)CO1 C(C(C)C)(C(O)C(=O)NCC(C)=CC(N1CC(S(N)(=O)=O)C1)=O)OC Cc1nc(C(=O)NCC2CCN(C(=O)C(F)C(C)(F)F)CC2)ccc1C#N N1(C(Cc2c(C)ncs2)=O)CCN(C(c2cc(C(C)C)ccc2C)=O)C2CCC12 Cc1cc(C(=O)NC2C=CC(CNC(=O)CC(C)C(C)C)C2)c(F)cc1F C(C(C(=O)NOCC1CCCC1)N(C)C)NC(c1c(C)n(C)cn1)=O c1(OC)cccc(OCC(=O)NCC(N2CCN(C(=O)CSC3CC3)CC2)=O)c1 CCCC(C(=O)NCC1(O)CCN(C(=O)CC2CCCC(C)C2)CC1)S(N)(=O)=O C#Cc1cc(C(=O)Nc2ccccc2C2CCCCC2)ccc1Cl c12ncc(Cl)cc1N2.N1(C(Cc2c(OC)cccc2)=O)CC2CC1CN2C C1(CCNS(CC)(=O)=O)CCN(C(=O)Nc2ccc(C(C)(C)O)cc2)CC1 N1(C(Cc2c(C)cnn2C)=O)C2CCC1CC(NC(=O)CN1CC=CC1)C2 C(=O)(C(F)CC(C)C)NCC(COC)NC(COC(C)=O)=O C(C(C)(C)C(=O)N1CCC(O)(CNC(=O)CCOCC2CCCO2)C1)N(C)C N1(C(CC(C)O)=O)CCC2OCCN(C(=O)CCc3ccn(C)n3)C2C1 C1(N(C(CCNC(C)=O)=O)C)CN(C(C23CCCC2(C(N)=O)C3)=O)CCC1O c1(OCCC(=O)NCCOC2CN(C(C3C(C)(C)C3(F)F)=O)C2)ccc(Cl)cc1 N1(C(C2(C)CN(Cc3cc(Br)cc(F)c3O)C2)=O)CCc2c(O)cccc2C1 N1(C(Cc2c(C)occ2)=O)CCCC2(C1)CN(C(C1(C(F)F)CCC1)=O)CCO2 N(C1c2ccccc2CC1NC(=O)C=CC)C(CC(=C=C)C)=O CCC(C)CC(=O)C(=O)N1CCC(C)C(CC(=O)NC2CCC(CCO)CC2)C1 C1(C2CCN(Cc3ccc4ccoc4c3)C2)(NC(c2c(C)ncs2)=O)CC1 Cc1cc(CNCCOc2ccc(F)cc2C)nc(Cl)c1Br c1(C(N(C(C)C(=O)N(C(C)CCC2CC2)C)C)=O)ccc(Cl)s1 N1(C(C=Cc2cncc(C)c2)=O)CC(C2CCCN(C(=O)CC(C)C)C2)C1 CC(Cc1ccco1)C(=O)N(C1CC1)CC1CCCN1C(c1ccc(CO)s1)=O C1(NC(CC=CCNC(=O)CC(C2CCC2)C2CCC2)=O)CC2CSCC2C1 C1(O)(C(N2CC(COC)(CNC(=O)CS(N)(=O)=O)C2)=O)CN2CCC1CC2 N1(C(C(C)C2CCCO2)=O)CCCC2(CCN(C(=O)C(F)n3cccn3)CC2)C1 C(=O)(C1=COCCO1)N1CC2C(CNC(C(C)(C)n3cc(Cl)cn3)=O)C2C1 C1(CC(=O)NC2(C3CCC3)CCC2)CC2(CCCC2)CO1 C1(C(=O)NCC23N(C(c4ncc(N(C)C)nc4)=O)CC(C2)C3)CCC2(CCC2)O1 c1(C(N(CC(O)CNC(C2CC2C#N)=O)C)=O)n[nH]cc1Cl c1(C(N2C(CN(C(=O)C(C)(C)F)C)COCC2)=O)ccc2c(c1)OC(F)(F)O2 N1(C(C2(OC)CC2)=O)CC2CCC1C1CN(C(=O)CCc3ncc[nH]3)CC21 C1(C(=O)OC)(CCNC(=O)NCCCCCNS(C)(=O)=O)CCC1 c1(CNC(=O)Cn2cnnn2)ccc(Cl)c(C(N2C(C(F)F)(C(=O)O)CC2)=O)c1 C#CC1CCN(C(c2ccc(CNC(c3ccc(C)cc3)=O)cc2)=O)C1 N1(C(C2(C)COC2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1C1CCC1 c1(C(=O)OC)cc(NC(C2C3CN(C(C4CCC(=O)N4)=O)CC23)=O)c(F)c(Br)c1 C(=O)(CC(CC)CCCC)NC(CC=C)CNC(c1cc(CO)oc1C)=O CCCCCCC(C(=O)NC(C)CCCNC(c1ccc(C)nn1)=O)NC(C)=O C1(CCC)CCN(C(=O)CCN(CCCO)C(C2(CC)CCCO2)=O)C1 C1(C(=O)NCC2C3CN(C(C)=O)C(C3)C2)CN2CCCC2CO1 CC(C)CCC(O)C(=O)N1CC=CC(C(N2CCC(N3CC=CC3)C2)=O)C1 C1(C(=O)NC(CCCNC(C2(CC(C)C)CC2)=O)C)CC(=O)N(CCN(C)C)C1 N1(CCC)CC(C(=O)NCC2C=CCN2C(=O)CCN2CCCCCC2)CC1=O Cc1nc(O)nc(C)c1C(N1CC2CCC2(CCNC(C2CSC2)=O)C1)=O Cn1cc(C(=O)NC(Cc2ccc(C)n2C)C(=O)O)c(C2CCCO2)n1 C1(C(=O)NCC(CN(C(CC)=O)C)O)CC2CC(C1)CS(=O)(=O)C2 C(=O)(CS(=O)(=O)CCO)N1CCC(CC)(NC(c2csc(C)c2C)=O)CC1 CCC(CC)CCC(=O)N(CCCNC(=O)C(O)CCC(C)C)CCO C(=O)(C1=NOC2COCC12)NC1(CNC(c2n(C)nc(CO)c2)=O)CCCC1(C)C CC(C)(CC(=O)NC(CNC(C1CC2CCCN(C1)C2)=O)CO)C(F)(F)F C(CCC(C)C)(C(=O)NC1CN(C(=O)C=C(C)Cl)CC1N=[N+]=[N-])NC(C)=O Nc1ccc(-n2cc(C(O)CC(=O)N3CCCC3C(=O)O)nn2)cc1 C(C(C)C(=O)NC(CO)C(C)n1cc(Br)cn1)NC(C1CN(C(=O)NC)C1)=O c1(C(N2CC(NC(CS(C(C)C)(=O)=O)=O)C(OC)C2)=O)noc2c1CCCCC2 CC1CC(NC(c2ncccc2N(C)C)=O)CN1C(C1CC1C1CC1C)=O c1(C(=O)NC2CC(C)(CNC(C3CC3Cl)=O)C2)ccc(Nc2ccccc2)cc1 c1(C(N(C2CC3CCCC(C2)N3)c2ncc(C)cn2)=O)nc2ccccc2[nH]1 C1(F)(CNC(CC2(OC)CCCC2)=O)CC2CCC(C1)N2C(=O)C(C)C(F)(F)F c1(C(N(CCC#N)CCOC)=O)cccc2c1ccn2CC(C)C c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2O)cc(F)c(Cl)cc1F C1(CC)CN(C)C(=O)CN1C(=O)CC1CCN1C(=O)C(C1CCC1)OC C(=O)(C1=CCCCC1C)N(CCN(C(=O)C(c1ccccc1F)C)CC)CC C12(NC(C3(NC(C(CC)NC(N)=O)=O)CSC3)=O)CC1COC21CCC1 c1(C(=O)NC(C2CCN(C(CCOCC)=O)C2)C)cc(C)nc(Cl)c1N c1(N(CC(CC)C)C)cc(C)nc(N2CCN(CCOC)C(=O)C2)n1 C1(CC(=O)NC(CC(C)NC(c2cccc(NC(C)=O)c2)=O)C)OC(C)(C)OC1=O C(=O)(C(F)(CNC(C1COCC(C)O1)=O)C(C)C)Nc1c(CC)nsc1 CC1(C)OCCN(C(=O)Cc2cccc(CNC3=C(C#N)CCC3)c2)C1C(=O)O N1(C(c2n[nH]c(CC)c2Br)=O)CC2CC(NC(=O)CC=CC(C)(C)C)C1C2 N1(C(C23C(CN(C(CNC(CCCCC)=O)=O)C2)C3)=O)CC2(C1)OC(=O)NC2C N1(C(c2ncnc3sccc23)=O)CCCC2(CCCN2C(=O)C(F)CC2CC2)C1 C=CC(C)(O)C(=O)NCCOCCC(=O)NC1CCCC(C(N)=O)C1 C(=O)(C(C)(C)n1ccnn1)NCCC(C)N(C(COCCC=C)=O)C C1(CNC(c2ccsc2)C)CC12CCC2 c1(C(c2nnnn2C2CCOC2)NCCCCC(=O)OC)ccc(C#N)cc1F C1(C(C)NC(c2cccc(Cl)c2)=O)CCN(C(=O)C(=O)NCC2CC2)CC1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC1CC(NC(C2(C#N)CCOC2)=O)C1 c1(C(N(CC(C)O)CCNC(=O)Cn2cnnn2)=O)cc2sc(=O)n(C)c2s1 C1(C(N2CC(=CCC)C2)=O)CN(C(=O)C(C)CSC)CC1OC C1(CNC(CN(C(C)=O)C)=O)CCC2CC1CN2C(=O)Cc1ccccc1 C12(C(=O)NCC(CC(C)C)NC(C3CCS(=O)(=O)N3)=O)CCCN(CC1)C2 C(C)(C1=CCN(C)CC1)NC(=O)NC(c1nc(C)c(C)[nH]1)(C)C C1(CNC(=O)C(O)Cc2ccccc2)CC2COCC2N1C(C1CC1(F)F)=O Cc1ccn(CC(=O)NC2CCCC(CNC(C3CC3(Cl)Cl)=O)C2)c(=O)c1 N1(CC)CCOC2(CCOC2C)C1.c12ccc(cc1[N+](=O)[O-])[nH]2 CC1CN(c2ncccc2S(=O)(=O)NC2CC3(CCC3)C2)CC1P(C)(C)=O c1(C(=O)NC2CN(C(C(=O)NCCC)C)C(C)CC2)cccn2ccnc12 C1(NC(c2ccc(OC)nn2)=O)CC(S(=O)(=O)c2ccccc2)C1 N#Cc1ccccc1S(=O)(=O)NC1(C#N)CCN(C(c2ncn(C(F)F)n2)=O)C1 N1(C(Cc2ccc(OC)cn2)=O)CCCN(C(C2CC23CCC3)=O)CC1CO CC1CC(NC(c2coc(COC(C)(C)C)c2)=O)CN(C(C2(CO)CC2)=O)C1 C1(C(N2C(C)CC(CNC(c3coc(Cl)n3)=O)C2)=O)CC2(C1)CC(C#N)C2 N1(OC(=O)CC2CCOCC2OC)CCN(CCc2snc(CCC)n2)CC1 c1(C(CC)C(=O)N2CC(NC(=O)CC3CC3(C)C)C2)ccc2c(c1)OCO2 Cc1ncc(C(=O)N(C(CC(F)F)C(=O)N2CCC=C(Cl)C2)C)c(C)n1 c1(CCC(=O)NC(C(C)NC(=O)Cn2ccnn2)C)ccccc1-n1cccc1 N1(C(C(C)Cc2ccccc2F)=O)CC2(C1)CN(C(=O)CCC(F)(F)F)CCO2 C1(C(=O)NCc2c(C(=O)OC)nco2)CC(C)CN(C(c2nnn(C)c2N)=O)C1 N1(C(C(=O)NC(C)C)=O)CCC(NC(c2ccnn2CCF)=O)C1(C)C Cc1nsc(NC(C2CCN(C(C3(C)CCNC3=O)=O)C2)C)c1C#N C1(CCCC)CN(C(C2C(C)C2(F)F)=O)CCN1C(c1csc(COC)c1)=O c1(CC(N2CC(SC(F)F)C2)=O)ccc2nc(-c3cnc(F)c(F)c3)sc2c1 N1(C(C(C)=C(C)C)=O)CC2CCCC2(NC(=O)CC2CCN(CC(F)F)CC2)C1 C1(CC)N(C(=O)C(C)C)CCC1(C)C.c12nc(c(N)s1)C(=O)NC2c1ccccc1 c1(C(c2nnnn2C2CCOC2)NCCc2cc(C)no2)nc(C)c(C)n1C Cc1cc(C(=O)CCC(=O)NCC(C(C)(C)C)NC(=O)C(C)N2CCC2)c(C)s1 C(CC(=O)NOCCN(C)C)N(C(CCN(CCC)C)=O)CC1CCCCC1 Cc1cc(C(c2ccccn2)NCC(Cc2ccc(Cl)cc2)C(=O)O)cc(C)c1 c1(C(=O)NCCc2cn(CCCC(=O)OCC)nn2)ccc2oc(=O)oc2c1 CC1(C)C(CC(N2CC(OCCC(=O)NCC(O)CF)C2)=O)C1(C)C N1(C(c2occ(C)c2)=O)CCC(C)(CNC(=O)CSCC(F)(F)F)CC1 c1(C(N2CC(O)(c3cn(C4CCOCC4)nn3)C2)=O)cc2ccccc2[nH]1 n1(C(C)C)cnnc1SCC(=O)NCC(F)CNC(=O)C(C)n1cccn1 N1(C(C2N(CC)CCC2)=O)CCCC2CN(C(=O)C(C3CC3)C3CC3)CCC12 N1(C(CCC=C=C)=O)CC(CNC(c2cccc(F)c2C)=O)C(C)(C)C1 C(=O)(C1COc2ccc(Br)cc21)NCC(CNC(c1ccncc1O)=O)O CC1(C)C(NC(=O)CNC(=O)CNC(=O)CC2CCCC(O)C2)CC1O Cc1cc(C(=O)N(CC(C)CNC(c2cnn(C(C)C)c2C)=O)C)c(O)nn1 C(=O)(C#CC1CCCC1)N1C(C)C2CC1C2NC(=O)CCS(C)=O Cc1cc(C(=O)NC(C2CCCN2C(=O)C(C)n2cncn2)C)nnc1O Cc1cc(F)c(C(N2CC3CC2CN(C(c2nccs2)=O)C3)=O)cc1Br C(C)(C(C(=O)NC(C)CCCNC(c1sc(C)cc1C)=O)N(C)C)OC Cc1ccnc(C(=O)NCc2cncs2)c1.c12csc(n1)NC2=O C=CCCC(C(=O)N1CCN(CCO)C(=O)C1)NC(=O)C(O)C1CCC1 CC(CCCNC(=O)CC(=O)N(C)C)NC(=O)Cc1sccc1Cl CS(=O)(=O)c1ccc(C(N2CC(NC(C3CC34CCOC4)=O)C2)=O)s1 C(CCC(C)(C)C(=O)NC(C)COC(C)C)NC(CC(CC)SC)=O C(CCC(=O)N1CCCC(CC2CC2)C1)(C(C)C)NC(c1c(CC)csc1)=O CCC(F)(F)C(C)(C)C(=O)N1CCC(CNC(c2ncc(Cl)cc2Cl)=O)C(C)C1 CC1CC(N(C(=O)CC2(C)CCN(C(c3cc[nH]n3)=O)C2)C)CCO1 c1(NC(c2c(C3CC3)cccc2F)c2n(CCOC)nnn2)ccc(Cl)nc1C N1(C(C(=O)N(CCCC)CC)=O)CCCCC2(CCN(C(C3CNC(=O)N3)=O)C2)C1 c1(CN2CCC(N(C(=O)C(C(C)C)NS(C)(=O)=O)CC)C2)cc(S(N)(=O)=O)c[nH]1 c1(C(=O)NCC2CCC3(CN(C(C(N)=O)=O)C3)O2)cnc2c(c1)NC(=O)CO2 C(N=c1ccn(CCC#N)[nH]1)(c1ccc(SC)cc1)c1nnnn1CCCF C1(C(N2CC(NC(C3CCC4CC3CO4)=O)C(O)C2)=O)CC2CCCC(C1)C2 Cc1c(C(N2CC=CC(NC(C3CC34CCC4)=O)C2)=O)ccc2c1CCC2 C1(C(=O)NCC(CC)N(C(=O)C(C)SC)C)CCN(C(C)C)CC1 C1(C)(NC(C2CCN(C(CC=CCC)=O)C2C(C)C)=O)CCC(C)(C)CC1 c1(-c2cn(C3CC(OCC)CC3O)nn2)cc2[nH]ccc2cc1Cl c1(-c2scc(C(=O)Nc3[nH]nnc3-c3ccccc3)n2)ccccc1Cl c1(C(=O)NCCC2(C(=O)NC3CC(O)C3)CC2)cccc(CC2CCC2)c1 Cc1nn(C)c(C)c1OCC(=O)NC1CC(F)(CNC(=O)CCCN(C)C)C1 C1(CNC(C2CC(OC)C2)=O)CN(C(=O)C(C)(F)c2ccon2)CC1(C)C C1(C(=O)NCC23CC(CN2C(=O)Cn2ncn(C)c2=O)C3)(CC)CCNC1=O C1(N(C(c2ncc(C(F)F)cn2)C(=O)NCC2CCOC2)C)CCC2(CC1)CC2 C(=O)(CCCCCCCC)NC1(CO)CCN(C(c2c(CC)nn(C)c2)=O)C1 c1(NC(=O)CCCCN2CCC(O)CC2)ccc(Cl)c(NC(C)=O)c1 N1(C(c2c(OC)nccc2)=O)CCC(C2CCN(C(=O)C(C)(C)CO)C2)CC1 C(=O)(CCCCC(C)=O)N1C(CC)C(C(=O)NC(C)CC2CC2)CC1 N1(C(CNC(C)=O)=O)CCC(NC(=O)Cc2cc(C)ccc2F)C12CCC2 C(=O)(C(C)(C)C(F)F)NCC(C)(C)CNC(c1ccnn1CC1CC1)=O N1(C(CNC(CCCCC)=O)=O)CC2CCN(C(C3CSCC(=O)N3)=O)CC2C1 c1(C(=O)NC2(CC=C)CCN(C(=O)Cc3nocc3C)C2)ncc(Cl)nc1Cl C1(C(=O)NCCCN(C(C)C)C(C2CC2(Cl)Cl)=O)COc2cc(F)ccc2O1 C1(NC(=O)CC2CCC2)CCC2(CC1)CN(Cc1cc(C(F)(F)F)n[nH]1)C2 C1(CC(=O)NC(C)C(C)NC(C2(CO)CCOCC2)=O)CC(C)(C)CO1 N1(C(CC2C(=O)NC(=N)S2)=O)CCC(C2(NC(C3CCC(=O)NC3)=O)CC2)CC1 Cc1cc2cccc(C(=O)NC3C4CN(C(c5ccccc5CO)=O)CC34)c2[nH]1 C(=O)(CC(C)CC(C)C)N1CC(C(=O)NCc2ccc(C)o2)N(C)CC1 C1(CC#C)(C(=O)NC2CC(NC(c3ccc(NC)cn3)=O)C2)CCCCC1 N1(CC)CCN(C(=O)CC2(C)CCN(C(c3cncs3)=O)C2)CC1C C1(OC)CCC(C(=O)NC(C)(C)CCCNC(=O)CCC2CCCC(=O)N2)CC1 N1(C(c2c(C)ncc(N)c2)=O)CC(NC(=O)C(F)n2ccnc2)CC2(CCC2)C1 C1(NC(C(C)(C)N(C)C(=O)OC(C)(C)C)=O)CC(CO)C12CCC2 c1(C(=O)NCCC2(NC(C34CSCC3C4)=O)CCCC2)cccc([N+](=O)[O-])c1 Cc1cc(F)ccc1C(CC1CC2(COC2)C1)NC(=O)Cc1ncccc1C#N c1(CNc2ccc(-c3c(N)nccc3)nc2)ccc(Cl)c(Cl)c1 Cc1nc2ccccc2n1CC(=O)NCC1CC(F)(CNC(c2cc[nH]n2)=O)C1 c1(COC(=O)NCC(C2CCC2)N(C)C)nsc(=N)[nH]1 c1(OC)cc(C(=O)NCC2(O)CC(CNC(C3(C(=O)O)CC3C(C)C)=O)C2)on1 c1(OC)cccc(CCNC(=O)C(=O)N(C)CCOc2cccc(Cl)c2)n1 N1(C(CCC=CC)=O)CCN(C(C2CCNC(=O)C2)=O)C(CCOC)C1 C1(CC)CN(C(CC)C(=O)NC(C2CC(NCC)C(OC)C2)C)CCO1 N1(CCNC(C2CC=CCO2)=O)CCc2c(ncn2-c2ccc(F)cc2)C1 C12(C(=O)NC3CN(C(C(C)NC(=O)NC)=O)CC3C)CCC(C(F)F)(COC1)C2 C(=O)(C(C)CC(F)F)NCC1CC(NC(Cc2ccc(OCC)cc2)=O)CC1O Cc1ccc(O)c(C(=O)NC2CN(C(=O)CSC(=N)N)CCC2C(F)(F)F)n1 C1(CN(C(=O)C=CC2CC2)C)CCCN1C(=O)CCC1CC1 CC1C(=O)CCC(C(=O)OCc2cc(F)c(Cl)cc2F)C1(C)C N1(C(c2nc(OC)c(C)s2)=O)CC2(CC(NC(=O)CC3CCCCC34CC4)C2)C1 c1(C(=O)OC)ccc(OC)cc1NC(=O)CCC(=O)NCC(C)SC.C(C)(C)O N1(C(c2ccc(SCCC)cc2)=O)CCN(C(C2CCC2C)=O)C(CO)C1 c1(C(N(C2CCN(C(C3(C)CC3)=O)C2)C)=O)cc2n(n1)CCOC2 c1(OCC)nc(C)cc(C)c1CNC(=O)C(=O)N(c1cccc(C)c1)C c1(C(=O)NC2(C)CN3CCC2CC3)nc(O)nc(O)c1N.C=C1CC2(C1)C(=O)C2 C(c1cn(C)nn1)=CC(=O)N(CC(C)N(C(CNC(CC)=O)=O)C)C c1(-c2[nH]nc(CCC(=O)NC)n2)noc(C2=NOC(C)C2)n1 c1(N(C(C2C(NC(c3nc(COC)oc3)=O)CC=CC2)=O)C)cc(F)ccc1C C1(C(C)NC(c2cccc(CNc3cc(C(F)F)nn3C)c2)=O)CN(C)CCO1 c1(C(=O)NCC(C)CN(C)C(C2(C)CCN(C)C2)=O)ncsc1S(N)(=O)=O S(=O)(=O)(c1ccc(O)cc1)NCC12C(CN(C(c3ncc(OC)cc3F)=O)C1)C2 C(=O)(C1=NN(C)C(=O)CC1)N(C1CCN(C2COCC2O)CC1)C Nc1c(C(=O)NCC2CN(C(c3c[nH]c4nccc-4c3)=O)C2)cc(F)c(F)c1F Cc1ncc2cc(C(=O)N(C3CCC(NC(=O)C4CC4)CC3)C)ccn12 c1(C(N2CC(N(C(c3cc(C(C)C)no3)=O)C)C2)=O)ccc2c(c1)CCCC2=O C1(CNC(C2N(C)CCCCC2)=O)CN(C(C2CC2C(F)F)=O)C2(CCC2)C1 C1(CCN(C(C(CN(CC)CC)F)=O)C)CCCCN1C(c1cccc(Cl)c1)=O N1(C(C2C(COCC)C2)=O)CCN(C(c2cnc(O)s2)=O)CC1c1nccn1C c1(C(=O)NC2CCCC(CNC(C3N(CC)CC3)=O)C2)c(OC)ccc(Cl)c1F N1(C(c2c(C)cno2)=O)CCC(NC(c2scnc2Cl)=O)C1c1ccccc1 N1(C(C(C)CN(C)C)=O)CCC(C)(C)C1C(=O)NC1CN(c2ncco2)C1 N1(C(CC(C(CC)C)NC(=O)C(C)(CO)OC)=O)CCCC2(CCCC2)C1 Cc1ccsc1C=CC(=O)NC1CCC(NC(=O)C(O)c2cnc[nH]2)CC1 N1(C(C=CCC)=O)CCC2(CC1)C1CC(C2(F)F)C(=CCCCCC)C(=O)N1 C(C(=O)NC1CN(C(=O)C=C(C)Cl)CC1CO)(C(C)C)NC(C)=O C1(C)(C(=O)NC(C)CN2CC=CC2)CCN(C(=O)Cc2cnoc2)CC1 O=C(C1(C2CCCC2)OCCO1)N(C12CC(Br)(C1)C2)CCSCc1ccccc1 Cc1cnn(CC(=O)NC(C)(C(=O)N(C(CF)CF)C)C2CCC2)c1 c1(CN(CC(N2C(CC)CCCC2)=O)C(C2CCC2)=O)cccc2[nH]ncc12 c1(C(=O)NCCCN(C(C(F)=CC)=O)CCO)ccc(-n2cncn2)cn1 C1(N(C(C(CC)=CC)=O)C)CCC2CN(C(=O)Cc3nccn3C)CC12 C1(S(=O)(=O)NC(c2ccccc2F)=O)(c2cn(CC(C)C)nn2)CCC1 C(=O)(C(C)(C)CCNC(=O)CC1CSC1)NC(C1CSC1)C C1(NC(c2cnc(C3(c4ccccc4)CCOCC3)[nH]2)=O)CCCC(F)(F)C1 N1(C(CCSCC(N)=O)=O)CCC(NC(=O)CC2CC(F)C2)C(O)C1 c1(N(c2ccccc2)C)cccc2cc(NC(=O)C(c3ccccc3I)N)cnc12 c1(Cn2cc(C3N(C(CNC(C(C)C)=O)=O)CCC3)nn2)cn(C)c(=O)cn1 c1(NC(C2CC(C)(C(N3CCCC(COC)C3)=O)C2)=O)cc(O)nc(C)n1 N1(C(C(N2CCCC(C)C2)=O)=O)CC(NC(=O)C=Cc2ncc[nH]2)CCC(O)C1 C(c1ccco1)=C(C)C(=O)NC1CC(OCC(=O)NCC2(C)CCCO2)C1 C(=O)(CC(C)(C)C(F)F)N(CC(C)CNC(=O)CC1(C)CC1(Cl)Cl)C C1(CNC(CN(C)C)=O)CN(CCCc2nnnn2C2CC2)CCCO1 C(=O)(CCCCCCn1cnnn1)NC(CCNC(c1c(C)cc(F)cn1)=O)C C(CCCCC(=O)N1CCC(OCC(C)C)C1)n1cc(-c2nc(C)sc2)nn1 C(=O)(C1=COCCC1)NC1C(CNC(c2cccc(C3(C)OCCO3)n2)=O)CC1 C(=O)(C(C)P(C)(C)=O)NCCC1(NC(Cc2c(C)ccnc2)=O)CC1 c1(C(=O)NC(CC=C)CNC(C2(C(C)(C)C)CCC2)=O)cnc2cccnc2c1 C=CCC(C)(C)C(=O)N1CCCC(N(C(=O)C=C2CCC(C)C2)CCO)C1 N1(C(=O)CC2CCCCCC2)CC2CCC(CNC(=O)C(F)(F)CO)(C2)C1 c1(C(N)=O)cccc(C(=O)N(CCCNC(=O)C=CSCc2ccco2)C2CC2)n1 N1(C(COCCOC)=O)CCN(C(c2ccnn2C)=O)CC1COC.C1C(=O)N1 CC(C)C(CCN(C(=O)CCN(C)C)C)NC(c1cc(-c2ccoc2)[nH]n1)=O C1(NC(=O)CCOC2CCC2)CN(C(=O)CC2CSC2)CC1C(F)F Cc1ccc(C(F)(F)F)c(C(=O)N(C2CC3CNC2C3)Cc2cc[nH]n2)c1 Cc1nn(C)c(Cl)c1C(N1CC2CC(C1)C2NC(c1ccnc(CO)c1)=O)=O O(NC(=O)C(CC(=C)Cl)NC(=O)C(F)CCC(C)C)C(C=C)C(=O)OC CC1CCN(C(=O)CCc2cc(Cl)no2)CCN1C(C1CCN(C(N)=O)CC1)=O c1(CCC(=O)OC)cnc(N2CCOC(C(O)C(=O)O)C2)nc1 C(=O)(C(F)(F)CO)NCC(c1ccc(F)cc1)NC(c1cc(SC)oc1)=O C1(c2ccc(F)cc2)(C(=O)NC(CC)CNC(c2[nH]ccc2C)=O)CCOCC1 C12(C(C)C)COC(C(=O)NCCC3CCCC(C(=O)N(C)C)C3)(C1)C2 C(=O)(C1=C(F)CN(C(c2cnsn2)=O)CC1)N(CC=C)CCC c1(NC2CC(O)(CNC(CC(CC)CN(C)C)=O)C2)ccc([N+](=O)[O-])c(OC)c1 c1(C(=O)NCC2(O)CN(c3nccc(CC)n3)C2)cc(F)cc(Cl)c1C c1(C(=O)NC2COCC2c2ccccc2)ccc(F)cc1C1CC1 C1(CNC(CS(CC)=O)=O)CN(C(c2ccc(C#N)cc2O)=O)CCC1(C)C CC1(C)CCN(C(C2CCC(C(N)=O)C2)=O)CC1CNC(=O)C#CC1CC1 c1(C(N2CC3CCN(C(C(CCC)C#N)=O)C3C2)=O)cc2cc(C)ccc2o1 C(=O)(C#CC1(C)CCCO1)NCC1(NC(c2cc(C3(C)CC3)on2)=O)CC1 c1(CC(=O)NCC(CO)NC(C2(CCCC)CC2)=O)cccc(OC(F)(F)F)c1 C(=O)(C1Cc2ccc(Cl)cc21)NC1(CO)CN(C(C2(C(C)(F)F)CC2)=O)C1 n1(CC)ccc(C(=O)NC2CC(C)(CNC(=O)C(F)(F)c3csc(C)c3)C2)n1 O=C1CN(C(=O)Cn2cncn2)C(C(=O)NC2CCN(CCCO)C2)CN1 c1(C(N(CC(C)NC(CCCCOCC)=O)C)=O)cc(OC)c2c(c1)OCO2 CC(C)C(F)(CNC(C1(C)C=CCC1)=O)C(=O)NCC(=O)N(C)C c1(CNC(CSCCC)=O)nnn(C)c1C(=O)NC1COCC1C(=O)NC c1(C(=O)OC2CCCC2)cc(C(F)(F)F)ccc1F.n12ccc(n1)NC(=O)C2 N1(C(CS(=O)(=O)NC)=O)CCC2(C1)CN(C(c1c(C)nsc1Cl)=O)C2 C1(O[Si](C[Si](C)(C)C)c2ccccc2C)CCON1S(=O)(=O)c1ccco1 c1(C(N(CC(CC)NC(c2cc(CCO)on2)=O)C)=O)cc2ncccc2[nH]1 CC(CC(N)=O)C(=O)NC1CC(F)(CNC(C2(CC3CCCC3)CCCC2)=O)C1 Cc1ccc(C(=O)NC(CNC(=O)CC(C)C2CC2)CC(C)C)c2c1CCC2 Cc1cc(N2CC3C(C(=O)NCCSC(C)C)C3C2)nc(C)c1 N1(C(C(C)OC)=O)CC(NC(=O)CC#N)C(O)C1 C1(CC(=O)NCCN(CCOC)C(c2ncsc2C)=O)CCC12CCC2 C(=O)(C(C)(O)CC(C)C)OC.C1C(C)(C)CC(=O)N1.C1(C)C(C)C(=O)N1 c1(C(CNC(C(CC)(F)F)=O)NC(=O)C2=CCSC2)ccc(Cl)cc1Cl S(=O)(=O)(c1cc(C(C)OC)ccc1C)NC(C(=O)OC)Cc1ccc(F)cc1 N1(C(C2(C)CC2(F)F)=O)CC2CC1CC2NC(C1(C(N)=O)CC1)=O C1(COC)(CN(c2nnc(-c3cccc(S(C)=O)c3)n2C)C)CC2CCCC2C1 CCCC(C)(O)CC(=O)N1CCC(NC(=O)CC2CC3CC3C2)C(CO)CC1 CC1CC(C(=O)NCCC2CN(C(=O)CCc3nccn3C)CCO2)CCN1C c1(C(N2CC3CC2CN3C(C2CC2c2cccs2)=O)=O)cc2n(n1)CCNC2=O N1(CC(=O)Nc2c(C)ncs2)CC2(CCCC2)OCC1C N1(C(C(C2(C)CCCCC2)C)=O)CC=C(CNC(=O)Cn2cccnc2=O)CC1 C12(C(N(C(CC)C)CC)=O)CCCC1CN(C(c1[nH]nnc1C1CC1)=O)C2 C1(C(=O)NC(C)(C(=O)NCC2CCC(C3CC3)O2)C2CCC2)CCC(F)(F)C1 N1(C(c2cnc(C)[nH]2)=O)CC2(CCCC2CC(=O)NC(c2c(C)noc2C)C)C1 C1(NC(c2c(C)n(C)nc2)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC1CO N1(C(CCC(=C)C)=O)CCCC(N(C)C(C2CC(Cl)(Cl)C2)=O)CC1 C1(CC(=O)N(CCC)C2CC2)N(C(=O)CC2CCCC23CC3)CCC1(C)C N1(C(CN2CCC(N(C3CC3)CC)C2)=O)CC2C=CC1CC2.c1ccccc1 CCCCCCCCC(F)C(=O)N1CC(C2(NC(C3C=CCCC3)=O)CC2)C1 N1(C(CC2C(CC)C2)=O)CCCC(O)(CNC(c2nccc(Cl)c2O)=O)C1 c1(NC(C2CC(=C)CN2C(=O)CN2CCCC2)=O)cc(OC(F)(F)F)ccc1O N1(C(c2cccc(CC)c2F)=O)CC2CCC(C1)N2C(c1[nH]c(=N)sc1CC)=O CCCCC(C)(F)C(=O)NC1CC1NC(=O)Cc1cncnc1O C1(C(C)NC(=O)CC2CCC3CC23)CCCCN1C(c1cscn1)=O c1(C(N2CCCC(F)(CNC(C3CC3C3CCC3)=O)C2)=O)cccc2sccc12 C1(CCC)NC(=O)CCN(Cc2ccc(Cl)cc2)N1CC(CO)C(F)(F)F N1(C(C2(SC)CCC2)=O)C2CCCC1CN(C(=O)C(C)SC(F)(F)F)CC2 N1(C(=O)CNS(CC)(=O)=O)C2CCC1C(NC(=O)C(=O)NC)C2 c1(C(=O)NCC(C2CCC2)NC(c2c(C)ccs2)=O)ccc(C)c(C)c1 Cc1cc(NC(=O)OC2CC(NC(=O)C(CC)C(C)O)C2OC(C)(C)C)nc(O)n1 c1(OC(c2ccccc2)C(=O)OC)cc(F)ccc1N.C1(=O)C(N)CCN1 c1(C(=O)NC(CN(C(=O)C(C)N(C)C)CC)C)sccc1C1CC1 c1(C(=O)NCC(C(C)(C)C)NC(CC=C=C)=O)cc(Cl)ccc1OC(F)F CN1CCCC12CCN(C(C1CCC3(CC3)N1C(c1nc(Cl)cs1)=O)=O)C2 c1(C(C)C)ccc(O)c(C(=O)N(CCCNC(=O)C(C)(F)F)C(C)C)c1 C1(CNC(CCCCCC)=O)C(C2CC2)CCN1C(c1cc(Cl)no1)=O C1(C#N)(C(N2CCC(CC=C)(NC(c3sc(F)cc3C)=O)C2)=O)CC2CC2C1 C12(CC(=O)NCCn3cccn3)CCC1CN(C(c1cccnc1O)=O)C2 CC1(C)CC(CC(=O)NCC2CC(NC(=O)CSc3n[nH]c(O)n3)C2)CO1 C(CCC(C(=O)N1CCC(OCCO)CC1)NC(c1cncn(C)c1=O)=O)OC c1(NCCNC(C2C(NC(c3cc(C(C)C)n[nH]3)=O)C2)=O)cccc2ccccc12 C1(CSC)CCCCN(CC(N2C3CCC2CC3)=O)C1 c1(C2(C(N(CCNC(CN(CC(C)(C)C)C)=O)C)=O)CCC2)ccc(Cl)c(Cl)c1 C1(C(=O)NCC=CCNC(C(C)CCc2cccc(F)c2)=O)CC12CCCCC2 c1(COCCCCOC(C)C)ccc(S(=O)(=O)N2CCOC(CCF)C2)cc1Cl C1(C(N(CCCCCNC(C(CC)(C)CO)=O)C)=O)CC(C)(C)OC1(C)C CC1CC(C(N2CSCC2C(=O)O)=O)CCN1 N1(C(C2CCC(C)(C)O2)=O)CCCC(O)(CNC(C2CC(F)C2)=O)C1 Cc1cc(NC(C2CCCC(C)C2)=O)cnc1F Cc1csc(C=CC(N2CC(NC(=O)C(O)C3CCCC3)C(C)C2)=O)n1 N1(C(c2cc(OC)no2)=O)CCN(C(=O)CC2CC(OC)C2)CC1 c1(C(=O)NCC(C)(C2CC2)NC(C)=O)cccc2c1CC(=O)N2C c1(C2C(C(=O)NC(CNC(CCOCCC)=O)CO)C2)ccc(F)cc1 N1(C(COCC(=O)OC)=O)CC2=C(C1)CN(C(c1c[nH]c(=O)c3ccsc13)=O)C2 c1(NCC2C(C)(C)OC(=O)C2)ccc2c(c1)CCC(=O)N2 CC1CCC(NC(c2coc(C(F)F)n2)=O)CN1Cc1ncc(Cl)n1C C(=O)(CS(=O)CCC(F)(F)F)N1CCC(C)(NC(CCSCC(N)=O)=O)C1 c1(CC(CNC(c2nc(-c3ccccc3O)cs2)=O)CO)ccccc1Br CCCCC(C)C(=O)NCC1CC2(CC(NC(=O)Cc3cscn3)C2)C1 c1(C(N(CCCNC(=O)C=C2CCC2)CC)=O)cc(C(=O)OC)cc(C(C)C)c1 C(=O)(CC1=NN(C)C(=O)C1)NC1C2C(NC(c3c(CC)scn3)=O)CC(CC2)C1 S(=O)(=O)(c1cccc(CNC(N2CC(CCCl)CC(F)C2)=O)c1)N1CCN(C)CC1 O=C(C=C(Cl)Cl)N(C1CC1)CC1(Cn2cc(-c3nccs3)nn2)CC1 C1(C)(NC(c2n(C)c(Cl)nc2)=O)CCCCC1C(=O)NCCCc1cncnc1 N1(C(Cc2ccc(OC)cn2)=O)CCC2C(CCCN2C(=O)C=Cc2cocn2)C1 C1(C(N2CCC(OCCNC(c3n(C)ncc3Cl)=O)CC2)=O)CCOC(C)(C)C1 CC(C)(CCNC(=O)OC(C)(C)C)C(=O)OCCNC(N)=O C1(CC)C(NC(C2(C)CS(=O)(=O)C2)=O)CCN1C(=O)CNC(=O)NC c1(OC)cc(CNC2CCNCC2c2ccnn2C)cc(OC)c1Br c1(C(N2CCN(C(C3(CO)CCCO3)=O)CC2CO)=O)cccc(Cl)c1Br c1(C(=O)NCC2(CSC)CC2)cc(CNC(=O)C=C(C)C)[nH]n1 CC1(C)C(CNC(c2ncc(C(F)(F)F)cc2Cl)=O)CCN1C(C1CC12CC2)=O C1(CNC(c2ccc(CSC)cc2)=O)CN(C(=O)Cc2ccc(C)s2)CC12CC2 N1(C(C2(C=C)CCC2)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1C C1(C(=O)NCC(C(C)C)NC(c2cccc(N)c2)=O)CC2C=CC1CCC2 N1(C(CC2ON=C(C)C2)=O)CC2(C=C(C(=O)NCC(F)F)CO2)C1 C1(NC(C(C)NC(N)=O)=O)CN(C(C2C(C)(C)C2(F)F)=O)C2(CCCCC2)C1 c1(OC)cc(C)c2cc(C(=O)NC3(CO)CCN(C(=O)OC(C)(C)C)C3)[nH]c2c1 C1(C)(CNC(=O)NC(c2ncc[nH]2)CC)CCN(C)C1 c1(CN(C(C2CC(Nc3cccc(OC)c3)C2(C)C)=O)CC)ccc(Br)cc1 C1(N(C(N)=O)C)CCN(N2CCCC(C(C)C)C2)CC1 c1(=O)n2ncc(c2N)[nH]1.C(C(F)(F)F)N(S(C)(=O)=O)C(C)C C1(C(=O)NCCCN(C(=O)Cc2cocn2)CC)COCCO1 C1(F)(NC(=O)OC)CCCN(C(=O)C(C)Oc2cc(C)cc(C)c2)C1 N1(C(Cc2nc(C)[nH]n2)=O)CC(CCNC(=O)C(C)(C)c2cnco2)C(C)C1 CN1C2CCC1CC(=CC(=O)NC1CC(NC(c3cc(N)c(F)cn3)=O)C1)C2 C1(C)(C(N(CC(C)NC(C2CC2c2cc[nH]c(=N)c2)=O)C)=O)CCC(=O)N(C)C1 N1(C(C=CC(=O)OCC)=O)CC2CCC1C(CNC(=O)CC1CC(C)OC1C)C2 CC(Cc1cnc[nH]1)C(=O)NCC1CCN1C(=O)Cn1cc(C(=O)O)cn1 N1(C(c2cncc(C)c2)=O)CC2(CCC2)CC1C(=O)NCc1c(C)n[nH]c1C C1(CC#C)(C(N2CCC(CCNC(=O)CN(C)C3CC3)C2)=O)CCCC1 C#CCCCCCC(=O)NC(C)(CNC(c1nccn1C)=O)C(C)C C(=O)(NNc1ncc2ccccc2n1)C(C)(C)C1CC1.CO C1(C(N2CC(O)(c3ccccc3)C2)=O)CCc2ccccc2O1 C(=O)(CCCC(=O)N(C)C)N1CC2C(CNC(c3c(C)cnn3C)=O)C2C1 Cc1cccc(CCC(=O)NCCC(C)N(C(=O)C(CO)NC(N)=O)C)n1 Cc1cccc(Cl)c1S(=O)(=O)N1CCC(CC(=O)NCC2COCCO2)CC1 C1(C(N(C2CCCC2)CC(C)NC(CC=CCC)=O)=O)CCCN(C(C)=O)C1 Cc1c(C(=O)NCC(C)N(C)C(c2ccc(CO)cn2)=O)cncc1Cl c1(C(C)C)nc(-c2nc[nH]n2)sc1C(=O)N(CCCN(C)C(C1(Cl)CC1)=O)C C1(c2cc(Cl)cc(OC)c2F)C2=C(N(C)C(=O)N1C)C(C)(C)N(C)C2=O CCC(CNC(=O)C(c1cccc(N)c1)O)(CC)NC(=O)C1=CCSC1 C(C(=O)NCCCN1CCC(NC(C2(CC(C)C)CC2)=O)C1)(C(C)(C)C)OC C=C=CCCC(=O)N1CC(C)(NC(C2C(C(=O)O)C2(C)C)=O)C1 C1(NC(=O)CC2COCCO2)CCCN(C(=O)CCc2cnoc2)C1 N1CCC(CCSC)CC1.O(C(F)(F)F)CC(=O)NCCCC1(SC)CC1 C1(CNC(Cc2c(C)nsc2)=O)CCC(C)CN1C(c1csc(CC(C)C)n1)=O Cc1c(C(=O)NC2CC(CNC(c3c(C4CC4)cnn3C)=O)C2)cnn1C c1(CC)occ(C)c1C(N1CCC=CC1C(=O)NCC(F)F)=O Cc1ccc([N+](=O)[O-])c(NC(C2C3CC2N(Cc2cccc(OCF)c2)C3)=O)n1 C1(NC(c2ccc(OC)cn2)=O)CCN(C)C12CCCN(C(C1CC(O)C1)=O)C2 c1(C(=O)NCC(C)CNC(C2(N(C)C)CC2)=O)cccc(C2CCCCC2)n1 c1(C(=O)NCC(C)NC(C2C(F)(F)C23CC3)=O)ccc(F)c(Cl)c1N CC1(CNC(C2(CF)CCN(C(C3CNC(=O)O3)=O)C2)=O)NC(=O)NC1=O N1(C(Cc2c(C)non2)=O)CCCC(C(C)NC(=O)C=Cc2cncn2C)C1 CCCC(=O)N(C)CCN(C(=O)C(C)O)C(C)C Cc1cccc(C)c1OCC(=O)NCC1(F)CCC(NC(=O)Cn2nccn2)C1 N1(C(c2ccc(C(C)=O)s2)=O)CCCCC1CN(C)C(c1cnc(C(N)=O)s1)=O C1(CC=C)(NC(c2sccc2C)=O)CCN(C(=O)Cc2cccs2)C1 Cc1nc(C(C)C)ccc1COC(C1(c2ccc(Cl)cc2)CC1C)=O C1(NC(CC2(C(=O)OC)CC2)=O)CN(C(=O)CCc2ccccn2)C2CCCCC12 C1(NC(CCOC(C)=O)=O)CC(C(=O)NCC2CC3CCC2O3)C1(C)C N1(C(c2cnc(C(=O)OC)s2)=O)CC(C2CN(C(C3CCC(C(N)=O)C3)=O)C2)C1 N(C(=NCC#Cc1cnn(C)c1)N(C)CC1CCOC(C(C)C)C1)C(C=C)C C1(C(=O)NCCCN(C(Cc2c(C)scc2)=O)C(C)C)CC(O)C(=O)N1 c1(C(N(CCCNC(c2cscc2Cl)=O)C2CC2)=O)csc(O)n1 N1(C(c2nc(C)[nH]n2)C(=O)Nc2ccc3c(c2)CCC3)CC2C(=O)NC(=O)C2C1 c1(CCN2C(CC(=O)OC)CCC2)ccc(Cl)nc1 C1(CC(=O)N(C2CCCC2(C)O)C)CCCC(NC(=O)CC2CC3(CC3)CO2)C1 c1(OCOC)ccc(C(=O)NC2CCN(C(C3CN(CC(C)C)C3)=O)C2)cc1 C(CC(CC)C(=O)N(CCC(=O)NCC(=O)N(CC)OC)C(C)C)=CC C=CCCCC(C1CC1)NC(=O)C(Cn1cncn1)NC(=O)C(C)n1cccc1 S(=O)(=O)(c1ccc(C(=O)N=c2cc(F)n(C)[nH]2)cc1)N(c1cccc(C)n1)C N1(C(c2c(CC=C)cccc2)=O)CC(C(=O)NC(c2nncs2)C)CC12CCC2 c1(OC)cc(C(=O)N(C2CCC(NC(C3(C)CC3F)=O)CC2)C)c(F)c(Cl)c1 c1(C(N(CC=C)C2CC2)=O)ncoc1CNC(=O)CC(C)n1cccn1 C=CCC(CC=C)C(=O)OCC1CCC(C)CO1 C(=O)(CC(C)CCC(=O)NCC(O)CNC(c1cnn(CC(F)F)c1C)=O)OC C1(F)(C(C)C)CCN(C(C2(C)CN(C(=O)CCCC3CCC3)C2)=O)C1 C(C)(CCC#N)(c1nnnn1CCOCC1CC1)Nc1ccc(CC)[nH]1 C1(NC(CC(=O)OC)=O)CCCCC1NC(=O)CSS(C)(=O)=O CCC(CC)(CCOC)C(=O)NCCCS(N)(=O)=O.c12cccc(n1)S(=O)(=O)N2 C1(C(=O)NCC(CN(C(C2(CCCC)CC2)=O)C)(C)C)CC2CC(O)C(C1)C2 C(CCC(C)(C)C(=O)N1CC(CN(C)C)C(C)C1)NC(C1=C(C)CCC1)=O CC1CC(CNC(=O)C(Cl)=CCl)CN1C(=O)Cc1cccc(O)c1 CC1(C#N)CC2(CC(NCc3noc4ccc(Cl)cc34)C2)C1 c1(-c2cn(CC(=O)NC(c3nnc(C(F)F)o3)C)nn2)ccc(C#N)cc1N C12(NC(c3ccc(OC)cc3)=O)CCCN(C(=O)COc3ccccc3)CC1C2 CC1(C)CCCCC(C(N2CC(NC(C3CC(F)C3)=O)C2)=O)C1 C12(C(=O)OC)CCCC1(C(=O)NCC(C)NC(=O)Cc1sc(=N)[nH]c1C1CC1)C2 C1(C(=O)NCC(C2CC(F)(F)C2)=O)CC(F)(c2ccccc2)C1 N1(C(C(C)N2CCCC2)=O)CCOCC1CC=CC(N1CC(O)(c2cc[nH]n2)C1)=O c1(CN2CCN(C(c3ncc(C(=O)O)cc3Cl)=O)CC2)c(Cl)cccc1B(O)O N1(C(C=CC(CC)=CC)=O)CCS(=O)(=O)C(CCNC(c2ccc[nH]2)=O)C1 N1(C(C2OCCN(CC)C2)=O)CC(C(N2CCCCC2C(=O)NC)=O)CCC1C N1(C(C)C)CC2CN(C(C3CCc4nc(C(F)(F)F)cn4C3)=O)CCN2C1=O C12(C(=O)NC(C(=O)OC)C)CC(CO)(CN1C(=O)Cn1cnc(=N)[nH]1)C2 c1(-c2c(OC)nc(OC)cc2)cnc2c(C(N3CCCC3C(C)C)=O)c[nH]c2c1 CC(F)(F)C(C)(C)CNC(=NCCF)NCC1CC12CCSCC2 N1(S(CCC)(=O)=O)CCCC(C(=O)Nc2nccn2C)C1 c1(OCC)ccc(CN2CCC2C(=O)NC(CCc2ccccc2)C2CC2)cc1C c1(CNC(C2C(NC(C34CC(COC)(C3)C4)=O)C2)=O)nc(C)c(C)nc1C C1(NC(c2c(OCC)n[nH]c2)=O)CCCC12CCN(C(=O)C(C)(CC)CO)CC2 C(C(=O)Nc1cccc(CSC(C)C)c1)(C(F)(F)F)c1ccc(C)cc1 n1(CC)nnc2c1CCC(C(=O)Nc1ccc(SC(F)(F)F)nc1)C2 Cc1scnc1C(N1CC(C)(NC(CC(n2ccnc2)C)=O)C1)=O c1(C(CC)C(=O)NCCC2CN(C(C)=O)C2)c(C)noc1C.C(=O)(C)NCC(F)F C1(NC(C2CCN(CC)C2)=O)CC2CN(C(c3cc(OC)cc(F)c3)=O)CC2C1 c1(COC(C)=O)nsc2ccc(Cl)cc12.c12cccc(c1)C=CC(=O)O2 N1(C(c2ncc(COC)s2)C(=O)NCC2CCCO2)CCCS(=O)(=O)CC1C N1(C(C(CC=CCC)C)=O)CCN(C(=O)CC2CCC(C(=O)OC)CC2)C(C)C1 C(=O)(C(C(C)C)SC)NCc1cc(C(=O)NC2CC(SC)C2)n[nH]1 c1(C(N2CCCC(CC=C)(NC(=O)CC(C)C(C)C)C2)=O)cc(Cl)c(N)cc1C CC1(CNC(c2scnc2C(F)(F)F)=O)CCCN(C(C2CC23CCCC3)=O)C1 n1(CCNC(=O)NC2CC(CC(C)C)OCC2)cc(C#N)ccc1=O c1(CC)oc2ccccc2c1C(=O)NCCCN(C(c1cc2n(n1)CCC2)=O)CC c1(NCCC(=O)NCC2C(OC)COCC2)nc(Cl)c(Br)cc1O Cc1noc2ncnc(NC(C)C(C3CCCCC3)NC(c3ncccn3)=O)c12 C1(C(=O)NC(CNC(c2ccn(C)n2)=O)C(C)(C)C)CC2(CCCCC2)S1(=O)=O C1(C2CCN(C(c3ccc(Cl)c(Cl)c3)=O)CC2)(NC(C2C(C)C2)=O)CCC1 N1(C(C(CCSC)NC(CC(=O)NCC#C)=O)=O)CC(O)C(C2CC2)C1 c1(OC)c(Cl)cc(C(=O)NC(C)CCNC(=O)CC2COCCO2)nc1Cl c1(C(=O)NCCN(CCCCCC)C(c2ccc[nH]2)=O)cc(O)c2sccc2c1 C1(CCC)CCCCC1C(N1CC(NC(c2ccoc2CC)=O)CC1C)=O C1(F)(C(=O)NCCC2CCN(c3snc(C(C)C)n3)CC2)CCCCC1 c1(CN2C(C(=O)Nc3ncc(I)cc3I)CC(=C)C2)ccc(OCC)c(F)c1F c1(CC(=O)NC(CNC(C2(CCC=C)CC2)=O)C2CCC2)cc([N+](=O)[O-])c(C)s1 C1(CNC(C(C)Cc2ccccc2)=O)CC2CCC1N2C(c1ncncc1N)=O c1(C(=O)NC2CCN(Cc3cn(CC(=C)CC)nn3)C2)ccc(Br)cc1Cl c1(C(=O)NCc2cc(C(=O)NCCC(C)SC)n[nH]2)cc(C)c(O)nn1 CC1(C)CN(C(C2CC=CCC2)=O)CC2(CN(C(C3CCC34CCC4)=O)C2)O1 c12ccc(nc1)CN2.C1(N(C2CCC2)CC=CC=O)CCCC1.C(CCC1CC1)O CCCCC(CC)CC(=O)N1CCC(NC(c2cc3c(s2)CCC3)=O)C(C)C1 C(=O)(C(CC)NC(C)=O)NC1CCC(NC(CC)=O)C1 C(CC(=O)NCCOC1CCN(C(C2CC23CC(O)C3)=O)C1)(C(F)(F)F)OC N1(C(C(C)CC2CC2)=O)CC2(C1)SCCC2NC(=O)CCCc1ccncc1 S(=O)(=O)(c1cccc(=NC(CC2CC2)CO)[nH]1)Nc1c([N+](=O)[O-])cccc1Cl C1(C(=O)NCC23CC2CN(C(=O)Cc2cnc[nH]2)C3)CC2CC1CC2(F)F C1(CC(=O)NC(CCOC)CNC(C2CC=CC2)=O)COCCN1C CS(=O)(=O)C1(C(N2CC=CC(NC(C3(C(F)(F)F)CC3)=O)C2)=O)CCCCC1 c1(C(=O)NC2CCN(C(c3c[nH]ccc3=O)=O)CC2CO)noc2c1CCCC2 c1(C(=O)NCC2C(NC(CC3C(C)(C)C3)=O)CC2)cn2ccnc2s1 c1(CN2C(C(N3CCC(CO)C(O)C3)=O)CC(O)C2)c(F)cc(I)cc1F CC1CN(C(C(=Cc2ccco2)C)=O)CCN(C(=O)C(C2CCCCC2)C)C1 c1(C(=O)NCC(CCOC)NC(=O)CC2CC2)cc([N+](=O)[O-])c(C)s1 C1(CC)(CC)CC(NC(=O)CC(C)(C)C)CN1C(c1cnn(CCOC)c1C)=O CC1CCN(C(=O)CC2CC3(C2)CN(C(C2CC=CC(O)C2)=O)C3)C(C)C1 C#Cc1ccc(C(N2CC3(CCN(C(c4scnc4C)=O)C3)C2)=O)cc1Cl c1(OC)cccc(-c2cccc(O)c2)c1C(=O)NC1CN(C(C)=O)CCC1O c1(C(N(C2CCN(C(c3snnc3CCC)=O)CC2)CC#C)=O)[nH]c(C)nc1C c1(C(N2C3CN(C(c4scc(C)c4)=O)C(C3)C2)=O)cnc(O)c2ccsc12 c1(C(N(CCN(C(C(CCC)C)=O)C)C)=O)ccc(-n2ccnc2)c(C)c1 O=C(C1=CCCOCC1)NC(C(=O)NC1CCOC12CCCC2)C1(O)CCC1 c1(NS(=O)(=O)CC=C(Cl)Cl)ccc2c(C(=O)O)cccc2c1 N1(C(C(=O)NCCOCCOC)=O)CC(NC(C2(C)CCCN2C)=O)CC(C)(C)C1 C1(C(=O)NCC2CC(NC(c3c(SC(C)C)nccc3)=O)C2)CC12CCCOC2 C1(NC(CSCC#C)=O)CCC(CNC(c2csc(C(F)F)c2)=O)C1 c1(CNC(CN(C(=O)CC2CC3CC3C2)C(C)C)=O)ccc(O)cc1F C1(CC)COC(C)CN1C(c1cccc(Br)n1)C(=O)NCCCC1CC1 C(C(C(=O)NC1CC1c1ccco1)n1cc(CC(C)(C)C)nn1)OCC c1(NC(c2n[nH]c3ccc(C(F)(F)F)cc23)=O)ccc(C(=O)O)c2cccnc12 S(=O)(=O)(c1c(OCc2c[nH]c3cccc(C(=O)O)c32)ccc(Cl)c1Cl)OC(F)(F)F N1(C(C(OCC)OCC)=O)CC(NC(=O)Cc2csc(C(C)C)n2)OC(C)(C)C1 C(CC(=O)NC1CCC(=O)N(C)C1)(C(C)(C)C)NC(c1c(C)c(=O)cc[nH]1)=O C(=O)(CN=c1[nH]c(C)cs1)NC1(CN(C(c2n(CC=C)ccc2)=O)C)CC1 C12(C(=O)NC(CC(C)C)C)CC(CO1)N(C(C1CC(C(C)C)C1)=O)C2 C1(NC(c2nc(C)oc2)=O)CCCCC12CCN(C(=O)CNC(N)=O)C2 c1(C(N2C(C)CC(CNC(Cc3c(C)ccs3)=O)C2)=O)cc2scnc2[nH]1 C1(C(=O)NCC2(Nc3ccc(C(=O)OCC)cn3)CCC2)Cc2ccccc2O1 c1(C(=O)NC2C(C)N(C(c3cnc(N(C)C)o3)=O)CCC2)cnc2n1CCOC2 c1(C(=O)N(C2CN(C(c3cncs3)=O)C2)C)ccc(CCCCC)cc1 c1(C(N2CC(CC)N(C(C3OCCN(C)C3=O)=O)CC2)=O)cc2cccnc2[nH]1 Cc1ccc(-n2ncc(C(=O)NCC(C(C)C)NC(=O)CC#N)c2C(F)F)cc1 Cc1cccc(C(=O)NCc2cn(CC(=O)N(CCCC(C)O)C)nn2)n1 N1(C(C(C)C2CC2)=O)CC(NC(C2SCCS2)=O)C(C)(C)C1 N1(C(c2c(CC)nc[nH]2)=O)CCC2(CCCC2NC(=O)CC2(N(C)C)COC2)C1 C1(CCC)CN(C(C2(CCF)CC2)=O)CC1NC(C1(C)CCCC1)=O C(C(O)CN=c1cc(Cl)nc(C(C)C)[nH]1)NC(CCCSC)=O C1(NC(C(c2cnn(C)c2)OC)=O)CCN(C(=O)CCOC(C2CCCC2)C)C1 CC1=NOC(C(=O)NCCCC2CCCN2C(c2ccccn2)=O)C1 c1(NCCCCNC(=O)NCCCCO)csc2cccc(F)c12 C1(CC(=O)NC(c2n(CC)cnn2)C)CN(C(=O)Nc2ccccc2)CCO1 C1(C(=O)OC(C)(C)C)CCN(C(=O)C(C2CC(F)(F)C2)O)C1.C(COC)(CO)OC C#CC1(C(=O)Nc2ccc(C(N)=O)o2)CCN(C(c2cn(C)nc2C)=O)C1 Cc1c(NC(=O)CCCNC(=O)Cc2cnnn2C)cccc1Cl C(CCC1CC1)(C(=O)NCCN1CCNC1=O)NC(c1cccnn1)=O c1(-c2nc(CCC)nn2CCOCC(F)(F)F)cc2ncccc2s1 c1(C(N2C(C)CC(CNC(=O)CN(C)S(N)(=O)=O)C2)=O)cc2cnn(C)c2s1 c1(CC)cc(C(=O)N(CC(=O)NC(CO)C(=O)OC)C2CCC2)n(C)n1 C(c1ccc(F)nc1)=CC(=O)NC1CC(CNC(=O)CNC(=O)C2CC2)C1 CCC(C)(C(=O)N1CCC(C(C)(C)CNC(=O)CC2CSC2)C1)C(N)=O CC1CCC(F)(C(=O)NCC2(F)CC(CNC(=O)CCS(C)(=O)=O)C2)CC1 c1(C(C(=O)NCC(=C)C)N(C2CC2)Cc2ccco2)cc(C)cc(Br)c1 c1(C(N(C2CCN(C(C(CCC)CCC)=O)CC2)C)=O)cc2oc(C)c(C)c2[nH]1 N1(C(CSSC)=O)CC(NC(C2CCCNS2(=O)=O)=O)CC12CCOCC2 c1(NC2CC(C)OC(C)C2)nccc(=NCCc2nnc(Br)n2C)[nH]1 c1(CC(=O)NC2CN(C(C=C(COC)C)=O)C(C)C2)ccnc(Cl)c1F c1(CNC(N2CCC(C)(CO)CC2)=O)cc2cccnc2cc1Cl C1(NC(c2c(C)nn(C)c2)=O)CCCN(Cc2ccc(-c3nn[nH]n3)cc2)CC1 c1(C(N2CC(CNC(C(C)(C)CO)=O)OCCC2)=O)cc(F)cc2nc(S)[nH]c12 c1(CC(=O)N(C)CC2(C)NC(=O)N(CC(C)(C)SC)C2=O)cnn2c1CCCC2 C(=O)(CC(C)(C)CC(=O)N1CC2(COC)CC1(CNC(=O)C(F)C(C)C)C2)OC C1(NC(CC(=C)C)=O)CCCN(C(=O)C(C)Cc2cccc(F)c2)CC1 CC1CCC=C1C(=O)NC(C(=O)NCCC1CC=CCC1)C1(O)CCC1 c1(-c2n(CC(C)C)c(N3CCCC(CC(F)F)C3)nn2)cc(C#N)ccn1 c1(C(N(C2(C(N(CCCOC)C)=O)CC2)C)=O)cnn(C)c1C(F)F C(CCC(C)CC(=O)N1CC2(CC(NC(C3(C#N)CC3(C)C)=O)C2)C1)=C(C)C C(N=c1cc[nH]c2cccnc12)c1c(-c2cccc(F)c2)n[nH]c1 c1(-c2ccccc2)ccc2nc(-n3cc(-c4cc5cnc(Cl)cc5s4)nn3)sc2c1 c1(C2N(C(C3C(C)C=C(C)CC3)C)CCC2)nc2ccccc2[nH]1.C(CSC)NC=O C1(CC(=O)NC2CCC(NC(=O)C3=NNC(=O)C3)CC2)CCCCCC1(F)F c1(CC(=O)OC)cccc(C(=O)NCC2CCCN(C(C3(Cl)CC3(F)F)=O)C2)c1 CC1(C)OCCC1C(=O)NCc1csc(C(=O)NCCc2nccs2)c1 C1(n2cc(CC3N(CC)CCC3)nn2)CCCN(C(=O)C(N2CCOCC2)C)C1 C1(CNC(C(CC)C)=O)CC2(CO1)CN(C(=O)C=Cc1cc(C(=O)OC)co1)C2 N1(C(CCN(C(c2cnc(C)n2C)=O)C(C)C)=O)CCC(O)(C(C)C)CC1 c1(C2C(CC(=O)NCC3CN(C(=O)C(O)C4CCCC4)C3)C2)ccccc1 C1(F)(C(=O)OC(C=C)C)CCN(C(=O)Cc2ccc(OC)cc2)C1 C(=O)(C(CC(F)F)NC(C1CC(CC)C1)=O)NC1C(CC=C)COC1 c1(C(N(CCCC(=O)NCC(CCC)C)C)=O)c(C)nsc1C C=CCCC(C)N=c1nc2c(ncn2C(C)C)c(N2CCOCCC2C)[nH]1 O=S1(=O)CC2CC2(c2nc(-c3ccccc3NS(=O)(=O)C(F)F)no2)C1 CC1CN(C(=O)CC2CN(C(C3CCSC3)=O)C(C)(C)C2)Cc2nncn21 O=C(CCCC1(NC(c2cnn(C3CC3)c2)=O)CCC1)NCCc1ncc[nH]1 N1(c2c(C)c(NCCCN(C)C3CC3)ncn2)CC(C)OC2(CCOCC2)C1 Cc1ccc2c(C(=O)NCCCN(C)C(c3cnn(CC(F)F)c3)=O)coc2c1 Cc1sc(-c2nc(C3CC3)no2)nc1C(=O)NC(C)CC1CCCCN1C c1(C2C(NCc3cc(Br)c(Br)s3)C2)cccc(Cl)c1.C12C=CC(C1)C(=O)NC2 Cc1c(Cl)ccc(C(=O)N(c2ncnn3cccc23)CCc2c[nH]c(=N)s2)c1F CCCCC(CC)C(=O)N1CCCC(NC(c2cccc(C(N)=O)c2)=O)CCC1 N1(C(C2CCN(C(C(C)NC=O)=O)CC2)=O)CC2CC3CC2C1C3 n1(CC(N2CC(CCNC(c3cnc(-c4ccccc4)[nH]3)=O)C2)=O)cnnc1O CCCC(C)(O)C(=O)NC(C)CN(C(=O)C(C)CSC(F)(F)F)C c1(C(N2CCCC(NC(c3cc(C)sc3)=O)C2C)=O)cc(=O)c2ccccc2[nH]1 CC(C)CC(C(=O)NOCCC(F)F)NC(C12CCCC1CCC2)=O.O(NC(C)C)C O(P(C)(=O)CNC(=O)CC1CC(C)N(C(=O)Cc2cn(C)cn2)C1)CC CC1CCC(CNC(c2cc(C3CC3)no2)=O)CN1C(c1c[nH]nc1Br)=O c1(C(=O)OC)nc(=NCC2CCCN2C(=O)C(C)CN(C)C)c(F)c(Cl)[nH]1 c1(C(=O)NCCCC(C)NC(c2c(OC)cccc2)=O)csc2c(F)cccc12 c1(C(N2CC3C(CNC(=O)Cc4cc[nH]c4)(C3)C2)=O)ccc2c(c1)C(=O)NCC2 c1(C(=O)NCC(CC(=O)Nc2cccc(C)c2C)OC)cc(F)cc(F)c1 CC(F)(F)CCC(=O)N1CCC1CNC(C1(CCS(N)(=O)=O)CCC1)=O c1(SCCCCC(=O)N2C(C)(C(NOCC)=O)CC2)cc(F)ccc1C C(=O)(CCS(=O)(=O)C1CCCC1)NCC1CCCN(C(C2(C)CC(C#N)C2)=O)C1 CN1CCC(O)(CC(=O)NCC2CCN2C(=O)C(C)(C)COC(C)(C)C)CC1 n1(CC)nc(C)cc1C(=O)NCCO.C(CCN=[N+]=[N-])CC#CCN C(CNC(C1(C(=O)N(C)C)CC1)=O)(CC(F)(F)F)NC(C1N(C(C)=O)CC(O)C1)=O C(=O)(C(CCC(C)C)NC(=O)CCC1CCOC1)N1C(CCC)CCC1 c1(C(=O)NCC2N(S(CCC)(=O)=O)C3C(C2)C3)cc(Br)ncc1OC c1(C(N2CC(CCNC(C(COC)(C)O)=O)C2)=O)cc(O)nc(Cl)c1 C(c1cccnc1)=C(C(=O)N(C(C)CNC(c1c(C(C)C)n[nH]c1C)=O)CC)C C(C)(C)(CC(=O)N1CCCCC1Cn1cc(CCC(C)(C)O)nn1)OC Cc1cn(C(C)(C)C(=O)N(CCCNC(C2CCC(=O)N2)=O)C2CC2)cn1 c1(C(N(C2CCN(C(C(C)NC(N)=O)=O)CC2)C)=O)cncc2[nH]ccc12 C(C(F)(C(=O)N1CC(NC(C)=O)C1)C(C)C)N(C)NC(C1(CC)CCCC1)=O C1(NC(=O)CCn2cnnn2)CN(C(C2CCSC2)=O)CC12CCS(=O)(=O)CC2 C(=O)(CC(C)CCC=C(C)C)NC1C(NC(c2c(C)ocn2)=O)CCOC1 C(CCC(C)NC(c1nscc1Br)=O)NC(C1C(CC(C)C)C1)=O C1(NC(C2(c3c(C)cccc3)CC2)=O)CC2CCC(C1)N2C(=O)C1=COCC1 c1(C(=O)NC2CC(NC(C3CC(CCC)OCC3)=O)C2)ccc2nnn(C)c2c1 CC1CN(C(c2ccnnc2)=O)CCC1CNC(c1ccc(=N)[nH]c1)=O C1(NC(c2c(CC)nccn2)=O)CC(F)CN(C(c2cc3n(n2)CCO3)=O)C1 c1(C(=O)Cc2c(C)nns2)cccc(F)c1C.c12cn(nn1)CCNC2=O c1(C(=O)NC(C)C(CO)NC(C2(O)CCC2)=O)cc(OC2CCCC2)ccn1 Nc1c(C(=O)NCC2CN(C(c3occc3Cl)=O)CCCO2)cccc1Cl C1(NC(C(C(C)NC(c2n[nH]c(C)c2C)=O)(C)C)=O)CC2CC1OC(=O)N2 N1(C(C2(OCC)CCOC2)=O)CC2CC1C2CNC(=O)CC1(CO)CCOCC1 C1(CNC(c2c(C)nc(C)o2)=O)CN(C(c2ccncc2)=O)CC(C(F)(F)F)O1 CC(C)CCN=C(NCC(c1cccc(F)c1)C)NC1CC1CC(C)C c1(CC(=O)NCC=CCNC(c2sccc2Cl)=O)cc(F)ccc1C(F)(F)F C1(OC(C(C)C)C(=O)NC2CCN(C)C2=O)C2CC3C1C3C2NC(=O)C1CC1 C(=O)(C(F)CC(C)(C)C)NCCOCCCNC(Cc1ccc(C)nc1)=O C1(CC(=O)OC)CCN(C(c2cnns2)=O)C1.C12CCC(C1)NC(=O)C2 N1(C(CNC(=O)OC)=O)CC(C(=O)N(C2CCC3(CCC3)CC2)C)CC(C)(C)C1 c1(N2CCC(OC)(CNC(=O)CC3C(=O)NN=C3C)C2)ccnc2ccnn12 c1(NCC(=O)NC2(c3cc(F)cc(F)c3)CC2)cccc(Cl)c1Br Cc1cc(C)c(C(N2CCC(CF)(NC(=O)Cc3cncs3)C2)=O)c(O)n1 C1(CC)CN(C(c2cnn(CC)c2)=O)CC1NC(C1(CF)CC(F)(F)C1)=O Cc1ccc(C(=O)NCC2CCN(C(c3nccc(Cl)c3F)=O)CC2C)cc1F c1(C(N2CC(NC(CC3CC(=C)C3)=O)CC2(CC)CC)=O)cc(C)cc(Cl)c1N CCC(C)C(CC(=O)NCc1ncc(C)s1)NC(C1CCCCO1)=O C1(NC(c2ncn(CC)c2)=O)CCC12CCN(C(C1CCCCC1(C)C)=O)CC2 N1(C(C(C=C)OC)=O)CC2CCC(C1)C(NC(=O)Cc1cccs1)C2 N1(C(c2n(C(C)C)ncc2)=O)CC=CC1(C)C(=O)NCCOc1cnn(C)c1 C1(C(C)=O)C(C(=O)NC2(C(=O)NCCC(F)(F)Cl)CC2)C1(C)C N(C1CCc2cc(CNC(=O)C3=NOC4COCC34)ccc21)C(=O)OC(C)(C)C c1(CCC(C)N(CC)CC)nccn1C.C1(=O)CCOCCOCCN1 c1(OCC)ccc(NC(=O)NC(c2cc(C)nnc2C)c2ccccc2)cc1Cl C(=O)(CCCCC(F)(F)F)NC1CCN(C(C(C)=O)=O)CC1C Cc1ccc(CCC(=O)NC2CC(C(=O)NCC3(O)CCC3)C2(C)C)cc1 C1(CN(C(CC(C)OC)=O)C)CCN(C(C2CC(F)(F)CS2)=O)CC1 C(C(C)C(=O)NC1CCC(CNC(=O)CC(=O)N(C)C)C1)SC C(=O)(CCCCC(C)C)NC(CCC)C(=O)N1CC(O)(c2cc[nH]n2)C1 C1(CCC(=O)NCC(CO)NC(C2(CCF)CCOCC2)=O)CCCC(=O)N1 c1(N(CCOCC(=C)C)C)nc2ccc(S(=O)(=O)CCN3CC=CCC3)cc2s1 c1(OCC)cc(C(=O)NC(COC)C(=O)NC2(C(C)C)CCC2)[nH]n1 Cc1cc(COCC(=O)NC2CC(C)(CNC(c3cnoc3C)=O)C2)no1 N1(C(C2(C#C)CCCC2)=O)CCCC(O)(CNC(=O)CC2C=CS(=O)(=O)C2)CC1 c1(OC)cc(Cl)c(C(=O)Nc2ccc(C(=O)NCc3ccc(F)c(Cl)c3)nc2)cn1 Cc1ccc(C(=O)NC2(CN(C)C(C3CC3c3ccn(C)c3)=O)CC2)n1C C(CCN(C(=O)C(C)C)CCCCC)(C(C)C)NC(C1(C)CC(=C)C1)=O c1(C(=O)NC2C(NC(C(C)n3ccnc3)=O)CCCC2)cc2c(nc1N)CCC2 CC1(CC(=O)NC2(C(=O)NCCc3ccncn3)CSC2)CCOC1 C(CC#CC(C)(C)C)NC(C#CCNC(C1(C)CCN(C)C1)=O)=O N1(C(C2(CCC=C)CC2)=O)CCC2CC2(NC(=O)CCn2c(C)csc2=O)CC1 c1(CC)oc2ccccc2c1C(=O)NC1CCC(NC(=O)CCCNC(N)=O)C1 c1(C(=O)NC(C)(C)CCNC(c2nncs2)=O)ccc(C2(C(F)(F)F)CC2)cc1 CCC(F)(C(=O)OC)C(=O)NCCN(C(=O)CCSC(F)(F)F)CCCN(C)C.OC C1(C(C)C)C(NC(=O)CCN2CCN(C)CC2)CCN1C(=O)C=CC1CCOC1 c1(C(=O)NCC2COCCN(C(C(C(=O)OC)(C)C)=O)C2)cc2cc(Cl)sc2[nH]1 C1(C(=O)Oc2ccccn2)CC2(C1)CC2F C1(NC(C2ON=C(C)C2)=O)CCN(C(C2(N(C)C(=O)OC(C)(C)C)CC2)=O)CC1 c1(NC(CC2(C)CN(Cc3cccc(O)c3)C2)=O)cncc(C2CC2)c1 N1(C(c2cc(Br)c(F)cn2)C(=O)NC2CCOC2)CC2CCC1C(O)C2O N12CCC3CCC(CC13)OC2=O.N1(C(C2(CC)CC2)=O)CCC(CO)(CN(C)C)C1 c1(C(N2CCC(NC(C3CC=CC3)=O)C(F)C2)=O)cc(O)nc2ncccc12 c1(OC)noc(C(=O)NCC2CCCCC2NC(c2ccncn2)=O)c1Br N1(c2c(COC)c(Cl)ncn2)CCC(C)C(NC(c2cc3cccn3cn2)=O)C1C C(=O)(C(CC(=C)C)NC(=O)CCC(=C)Br)NCC1(C#C)CCCC1 Cc1ccc(CCOC(c2csc(NC(=O)Oc3ccc(F)cc3)n2)=O)cc1O Cc1cc(C(=O)NC2CC(O)CN(C(c3cccc(Cl)c3)=O)C2)nc(C)n1 C1(C(=O)NCC2(N(C)C)CCC(C)C2)CCCC2(CCCCC2)C1 N1(C(C2CCC(CC)O2)=O)CC2CC(C1)C2NC(c1ccccc1SC)=O N1(C(c2nnn(C(C)(C)C)n2)=O)CC(F)(F)CC1CNC(c1nn[nH]c1Cl)=O C(N=c1cccc(S(=O)(=O)NC2CCCN3CCCCC23)[nH]1)c1c(OC)c[nH]n1 C1(NC(C=Cc2ccc(SC)s2)=O)CC(NC(=O)CCC(C)(C)F)C12CCC2 Cc1cc(C(=O)OC(C)(C)C)ccc1NC(c1cocn1)=O.C12CCCC1NC2 N1(C(C2(C)CC=CC2)=O)CC2CCC1C(CNC(=O)CC1CCC3CC13)C2 C(=O)(CC(F)(F)F)N(CC)CC1CCN(C(=O)COc2ccccc2C(N)=O)C1 N1(C(c2cc(Cl)c(OC)c(Cl)n2)=O)CC(C)(CO)Oc2ccccc21 c1(OC)c(C(N2C3CCC2CN(S(=O)(=O)CC#N)C3)=O)cccc1[N+](=O)[O-] c1(CC(C(=O)N(CCC(N)=O)CC)NC(C2CCS2(=O)=O)=O)ccc(Cl)cc1Cl C(c1cnc[nH]1)=CC(=O)NCC(C)CNC(C1CC(F)(CO)C1)=O N1(C(c2cnc(=N)[nH]c2)=O)C(CC(N2CCC(C3(C)N=N3)C2)=O)C2CCCC12 c1(N(CC#CCCCO)C)cc(C(F)(F)F)ccc1N c1(C2(C(=O)NCC3CCN(C(C4CCCCO4)=O)C3)CCC2)ccc(Cl)c(F)c1 C1(CCC)CN(C(=O)Cn2cccc2)CC1C(=O)NCC(C)CCC C1(CC)CN(C(=O)C(O)CC(F)F)CCN1C(C1(NCCOC)CC1)=O c1(C(=O)NC(C(=O)NC(c2noc(C)n2)CC)CC2CCC2)cc(C)nc(C)n1 C(=O)(CCC(C)(F)F)NCC1(OC(F)(F)F)CCN(C(CCN(C)C)=O)C1 c1(OC)ccc(CC(=O)NCCCCN(C)C(c2sc(F)cc2C)=O)cn1 Cc1nc2cc(C(=O)NCC3CN(C(=O)C(=O)NC4CC4)CCC3C)ccc2o1 c1(OC)cnc(CN(CC(C)NC(c2cnc(-c3cnn(C)c3)s2)=O)C)nc1 Cc1n[nH]c(C)c1CC(=O)N(C1CCC(CNC(c2nnn(C)c2C)=O)CC1)C C1(NC(c2cnn(CCO)c2)=O)CC(O)CN(C(c2cc(Cl)ccc2Cl)=O)C1 N1(C(CCCNC(=O)NCC#C)=O)CCC(N(C(c2ccsn2)=O)CC)C(C)C1 CC1CCC(Cl)=C(C(=O)NC(C)CNC(c2cc(C(C)(C)C)nn2C)=O)C1 c1(CNC(CCOCC#C)=O)ccc(OCCC(=O)NC(C)(C)C)nc1 Cc1cc(Cl)c(C(N2CCC(CCNC(=O)C(N3CCNC3=O)C)C2)=O)cc1N C1(CC#C)(C(N2CC(N(C)C)CC2C)=O)CCN(C(c2ccc(CC)o2)=O)C1 Cc1cc(N2CCC(NS(=O)(=O)C3CC3)CC2)nc(=NCCc2csc(Br)c2)[nH]1 c1(C(=O)NC(CNC(c2c(CC)c[nH]n2)=O)CO)cc(C#N)ccc1Cl c1(CC(=O)NCCCN(C(c2n[nH]c(CC)c2Cl)=O)C(C)C)c(C)nn(C)c1C CCCCCCCCC(C)C(=O)NC1CC(NC(c2ccc(C(C)F)cc2)=O)C1 N1(C(c2ccc(F)cc2)=O)CCC2C(CCCN2Cc2ccccc2)C1 CC1CCC(O)(C(=O)NC2CCCN(C(c3ccn(C(C)(C)C)c3)=O)C2C)CC1 CC#CCC(C(=O)N1CC(O)CC1CC)NC(c1cccc(C)c1F)=O C(C(CO)C(F)(F)F)NC(c1cc(CNC(c2ccc(OC)o2)=O)on1)=O C1(CNS(CCOCC)(=O)=O)C2CCC1CN(C(c1ccccc1)C)C2 C(c1c(F)cccc1F)=CC(N1CCC(C(C)NC(c2ccnc(S)c2)=O)C1)=O Cc1ccn2c(C(=O)NC(C)CCCNC(=O)C(C)n3cccn3)cnc2c1 c1(C(N2C3CCC(NC(CN(CCC)C)=O)C(C3)C2)=O)cn(C)c(=O)n(C)c1=O c1(C(=O)NC(C2CN(C(=O)C=CC3CCCC3)C2)(C)C)cnc2n1CCC2 Cn1nc(CNC(=O)C(CO)N(C)C)cc1C(=O)NCCC(Cl)Cl CC1CCc2[nH]c(=NCC3CCCC(C)(C)O3)[nH]c(=NCC#CC3CC3)c2C1 C1(NC(=O)CCCn2ccnc2)CC2(C1)CN(C(c1cc(F)cnc1O)=O)C2 C1(NC(C(CC)C)=O)CC2CC(NC(c3ccncc3Cl)=O)C2C1 c1(CN(C)C(C2CC2C2CCCO2)=O)cccc(CNC(c2csc(F)c2)=O)c1 CCCCC#CC(C)(C)NC(C1CN(C(=O)C(C)(C)C(C)O)CC1CCC)=O c1(Nc2cc(NCC3(C(C)C)CCCC3)ncn2)ccc2sccc2c1 c1(OC)cc(F)ccc1S(=O)(=O)N(c1ccc(C#N)cc1)CC(C)C c1(C(N(CCCNC(=O)CC2COC(=O)C2)C)=O)[nH]nc2c1COC2(C)C c1(OC)ccc(C(=O)NCC(N2CCCC(CNC(=O)CC(F)(F)F)C2)=O)cc1 c1(CC(=O)NCCC2N(C(C(C)C3CC3)=O)CCSC2)cc(O)ccc1Br C1(CCC(=O)NCC23CC2CCN3C(=O)CC(F)(F)Cl)CCC(O)CC1 c1(C(=O)NC2(C3N(C(c4c(C)coc4)=O)CCC3)CC2)cc2n(n1)CCOC2 CC(C)(CCCNC(=O)CSc1ccccc1Cl)NC(=O)CCC1CCC1 c1(C(=O)NCCC(C)N(C(C2(C=C)CC2)=O)C)ccc(NS(C)(=O)=O)cc1Cl CCC(C(=O)N(C)CC1(NC(c2csnn2)=O)CC1)SCc1ccccc1 C1(C2CN(C(=O)CN(C)C(c3cccnc3)=O)C2)(NC(C(CC)OCC)=O)CC1 CCC(CC)C(=O)NCC(C)(CNC(=O)C(CC1CCC1)OC)NC(COC)=O C(C)(C(C)NC(C1(SC)CN(C(=O)CC2CCCSC2)C1)=O)(C1CC1)OC CCCCC(=O)C(=O)NC1CC(O)CN(C(=O)CC2(COC)CC2)C1 c1(C(=O)NCCN(C(CCOC)=O)CC(C)O)ccnc(C)c1O c1(C(N(C2(C(N3CC(CN(CC)CC)C3)=O)CC2)C)=O)cc(C)sc1N N1(C(=O)OC)CCCC2C1CCCN2C(c1c[nH]nc1CCOC)=O C1(C(N2CC(O)(CNC(=O)CNC(C3CCC3)=O)C2)=O)CCn2ccnc2C1 c1(CCC(N2CCN(C(=O)COCC(F)F)C3CC23)=O)c(Cl)cccc1Cl C1(NC(=O)CN)CCN(OC)CC1.CCCC1C(=O)N1 C1(C(=O)NCC(N2CCOCC2)C)CCN(C(C2CC(F)C(=O)N2)=O)C1(C)C CC(=O)CCCC(C)C(=O)NC(C)(C)CCCNC(C1CCn2cnnc2C1)=O Cc1ccc(-n2nc(-c3ccc(F)cc3)nc2-c2cnn(C)c2Br)cc1 N1(C(C(C)O)=O)CC2CCCC1C2CNC(c1ccc(Cl)c(F)c1)=O CC1(C)CC(NC(=O)CC(O)C2CCCC2)CN(C(C2(C)CC(C#N)C2)=O)C1 N1(C(c2cc(C)[nH]n2)=O)CCC(C)(CNC(=O)CCC2CCCCC2)C1 c1(N2CCCC(CCC=C)C2)ccncc1S(=O)(=O)NC1CCCN1C(C)C O=C(CS(=O)CCC(F)(F)F)NCC1(F)CCN(C(C2CCS2(=O)=O)=O)CC1 C1(C(N2CC(CC(C)(C)CNC(c3cc[nH]n3)=O)C2)=O)CCOCC1(C)C C1(C(=O)NCCC2(O)CN(C(CN3C(C)CCC3)=O)C2)CCS(=O)(=O)C1 C(C(=O)NCC1(C(=O)N(CC(C)C)CCOC)CCCO1)(C(C)C)OC C1(N)(C(=O)NC(C)CC2CCC2)CCCN(C)C1 C1(N(C(c2cc(C)nn2C2CCC2)=O)C)CC2CCC1CC2 C(C(C(C)(C)C)NC(C1(n2ccnn2)CC1)=O)NC(C(C)Cc1cnc[nH]1)=O C(=O)(CCC(=O)NCCN1CCC(NC(C)=O)CC1)NC1C(C)(CC)C1 N1(C(CSCCC)=O)CCC2CN(C(=O)CCc3ncccc3C)CC2C1 C(C(O)CC(=O)NCC1CCOC1)NC(c1cc(C)[nH]c1)=O c1(C(=O)NC2(CNC(c3c(CC)nc(C)[nH]3)=O)CC2)cc(F)ccc1F C(CN=C(NC(c1ccco1)C)NC1COC2CC1C2)OC N1(C(C2C(C)C2)=O)CC2(C1)SCCC2NC(=O)CC1NC(=O)NC1=O O=C(CCCCN1CCCC1)NCC1(F)CN(C(=O)Cc2cnccc2Cl)C1 c1(C(=O)NCC2(NC(c3cnn(CCCF)c3)=O)CC2)cc([N+](=O)[O-])cnc1O C(=O)(C1=CCCC1(C)C)Nc1cccc(NC(c2cnn(C)c2N)=O)c1 c1(C(N(CCNC(=O)C(F)(F)c2nccn2C)CC)=O)cnc2n1CC(C)CC2 C1(CCOC)CN(C(c2cnn(C)c(=O)c2)=O)CCN1C(C1CCCCS1)=O n1(CC(=O)N(CCOC2CCCCC2)CC)ncc(Br)n1 C1(NC(CC2C(C)CCN(C(c3cnc(=N)[nH]c3)=O)C2)=O)CC2CC1CC21CC1 CCCC(CC(C)C)C(=O)NCC1CCC2(CN(C(=O)C(C)N(C)C)C2)O1 CCC(C)(C#N)C(=O)N1CC2CC1CN2C(=O)Cc1cc(C(C)C)no1 N1(C(c2cc(C)no2)=O)CC(F)CC1CNC(=O)C(C)c1ccon1 c1(C(=O)NCCOCCCNC(C2OCC(C)(C)C2)=O)cccn2c(O)nnc12 c1(N2CCCC(CN(C)C)C2)nc(NCCCc2ncco2)c2c(ncn2C)n1 N1(C(C23CC(OC)C2C3)=O)CC2CC1(CNC(c1c[nH]nc1C)=O)C2 C1(C(=O)NC(C2CCN(C(=O)CC(C)(C)C)C2)C)CS(=O)(=O)CCO1 N1(C(c2nnn(C(C)(C)C)n2)=O)CCC(C(F)F)(CNC(c2nonc2N)=O)C1 c1(CNCc2ncc(OCC)cn2)c(C)c(C)c(C)c(C)c1C c1(NCCNC(N(C(C)NC(=O)CC(C)(C)C)CC)=O)c(S(C)(=O)=O)cnn1C CCC(O)C(F)(F)C(=O)N1C2CCC1CN(C(=O)Cc1cccc(SC)c1)C2 C1(=O)CCCCNC(=O)C2(CCC2)CCN1.C1(NC(C)(C)C)CC1OC.COC Fc1ccc(CNC(C2CCN(Cc3cc(C4CCOCC4)on3)C2)=O)cc1 c1(C(N2C3CN(C(C(CC)OC)=O)C(CC3)C2)=O)cn2c(n1)C(=O)N(C)CC2 C1(NC(CCC=CCC=C)=O)COCCC1NC(=O)Cc1cnccn1 C(CCC(=O)NC1CC(NC(C2(C(C)C)CC2)=O)C1)N(C(C)=O)C c1(C(N2CCCC(N(C(c3c(C)nco3)=O)C)C2)=O)cc2cc(F)cc(F)c2o1 C=CCCCC(=O)N1CCC(CN(C)C(c2ccc(OC)s2)=O)CC1 N1(C(C(C(C)O)(F)F)=O)CCC2CN(C(c3n[nH]c4cccnc34)=O)CC2C1 c1(CCC)nccc(N2CCN(CC(n3cc(C(C)(O)CC)nn3)C)CC2)n1 N1(C(C2(C)CC3(CCC3)C2)=O)CCOC2(CCCN(C(C3(O)CCOC3)=O)C2)C1 c1(-n2ccc(C)n2)cc(C(=O)N(C23CCC(C(=O)OC(C)(C)C)(C2)C3)CC)c(C)o1 C1(NC(C2C(C)C2)=O)CCCN(C(=O)CCCN(C(C)(C)C)C2CC2)C1C Cc1ccc(-c2nc(C(=O)NCC3CC3NC(=O)C(c3ccccc3)O)cs2)o1 C1(CC(N2C(C(C)(C)NC(CSCC#C)=O)CCC2)=O)SC(=N)NC1=O c1(OC)ccc(Br)c(F)c1NC(=O)C(C)ON1CCC(c2ccc(CO)cc2)C1 N1(C(=O)CC2CC2)CC2(C1)CN(C(C1CCC3(CCC3)CC1)=O)CC2CO C(=O)(C1CCCc2cncn21)N1C(CN(C)C(c2cccc[n+]2[O-])=O)COCC1 c1(C(N(C(CC(=O)OC)C)C2CC2)=O)nn(C)c(C2CC2)c1C.C12CN(C1)C(=O)O2 C(CC(O)CC(=O)NC1CC12CCCC2)SC c1(N2CCC(N(C(=O)CCC3CCCCO3)CC)C2)ccc([N+](=O)[O-])c(C#N)c1 N1(C(C2C(CC)CCO2)=O)CC(C)(C)CC1CC(=O)NCC(C)(C)O c1(C(=O)NCC2CCN(C(c3c(C)ncnc3)=O)C2)nc(C(F)(F)F)ccc1N CCCC(C(=O)NC1CC2CC(C1)N(C(c1conc1C(C)C)=O)C2)S(N)(=O)=O C1(C(=O)NCC(CCCC)NC(=O)CCCCC(C)C)CC12CCC(C)(C)CC2 N1(C(C(CC)(C)CC)=O)CC(C)CN(C(=O)Cn2cc(C3CC3)cn2)C(C)C1 C1(C(=O)NC2CC(C#C)C2)(NC(c2cnn(C3CC3)c2)=O)CCN(C)C1 Cc1nc2cncc(C(N3CCC(N(C)C(c4cc(Cl)n[nH]4)=O)C3)=O)c2[nH]1 N1(C(C2(C)CC2(Cl)Cl)=O)CCC2CN(C(=O)C=Cc3cnc[nH]3)C2C1 C1(C2CCC2)(CNC(C=CCC)=O)CCN(C(=O)C(C)CCCOC)CC1 C(CC(O)C(=O)NC1CC(C)(NC(C2CC(C)(O)C2)=O)C1)SC C(C(=O)O)(C1=CCC2CC2C1)NC(C(CC)(C)C)=O c1(-n2c(CO)nc(C(CC)C)n2)cccc2ncccc12 N1(C(c2ccc(OCP(C)(C)=O)cn2)=O)CC2(CCC2)C2COCC12 C1(C)(C(N2C(CC(C)C)CNCC2)=O)CC12CCN(CC1CCCOC1)CC2 Cc1noc(C)c1CNC(C1CSCCN1C(C1CCC2(CC2)C1)=O)=O C1(CN(C(=O)C(=O)NC(C2CCCCO2)=O)C)C2CN(C(=O)OC(C)(C)C)CC12 Cc1nc(O)ccc1C(=O)NC1(CNC(=O)C#CC2(C)CC2)CCOC1 Cc1nc(C(C)C)oc1C(=O)NCC(C)NC(c1cnc(-c2ccc(Cl)cc2)s1)=O c1(C(=O)NC2CC(C(=O)Nc3c(C(=O)OC)c(C)sc3)C2)ccc(F)cc1I c1(C(N2CC(CNC(c3coc(-c4cccs4)n3)=O)C2)=O)ncn2c1COCC2 C(=O)(C(C)CC(F)F)N(C1CCN(C(=O)CC(=O)OCC)C1)CC c1(N2CC3C(NC(=O)C(O)CC4CCCCC4)C3C2)cc2nncn2cn1 C(=O)(CCCC(CO)(CO)CO)N1CCC(C#C)(O)C1.C1(=O)C(CC(C)CC)N1 c1(CC)cc(C(N2CCC(NC(=O)C=C3CCC(C)C3)C(F)C2)=O)ccc1O C1(CNC(C2(CC(=O)NC(c3ccnn3C)CC)CC2)=O)CCC(C(=O)OC)O1 c1(CSC)ccc(C=CC(=O)NCC(C2CCC2)NC(C2(CF)CC2)=O)cc1 CCC(CNC(=O)C(F)C1CCC1)(CC)Nc1nnc(C)o1 CC1C(NC(c2nsnc2O)=O)CCCN1C(c1cnnn1C1CC1)=O C1(NC(Cc2nnc(C)o2)=O)CCC12CCN(C(c1ccc(F)c(Br)c1)=O)CC2 C(C(C)(C)CS(=O)(=O)NC1CC(OC(C)C)C1)OC C1(C)(CNC(C(NOC)=O)=O)CCCN(C(=O)CCc2c(F)cccc2F)C1 C=C(C)CN=C(NCc1ccccc1)NC1CC(OC)C12CCC2 c1(C=O)cc2ccccc2[nH]1.C(=O)(C(C(C)C)C1CCC1)N(CCC)CCN CCC(C)(C(=O)NC1CC2CC1CN(C(c1c(C)ncnc1O)=O)C2)C(N)=O C1(CNC(c2c(CC)occ2C)=O)CCN(C(=O)CS(=O)(=O)NC)C12CC2 Cc1ncn(-c2ccc(NCc3c(Br)cnn3C3CC3)cc2)c1C C1(C)(C(C)=O)CCN(Cc2cn(CC3CCN(C4COC4)CC3)nn2)C1 c1(C(N2CC(C)C(CNC(=O)COCCO)C2)=O)nc2c(s1)CCCC2 N1(C(CC2OCCN(C(CC=CCC)=O)C2)=O)CCC(F)(C#N)C1 n1(C(C)C)cc(-c2nc(CS(C)(=O)=O)nn2CCF)ccc1=O c1(C(=O)NC(C)(CNC(=O)CO)c2cn[nH]c2)cccc2ccc(Br)nc12 c1(C(C)=O)cc(C(=O)N(C)CCNC(C2CCC3C2C3(F)F)=O)ccc1O N1(C(C=CC)=O)CCCCC2(C1)CN(C(=O)COc1cccc(OC)c1)C2 N1(C(C=CC=CC)=O)CCN(C(C2CC3(C2)CC32CC2)=O)C(CO)C1 c1(CC(N2CCC(C(C)(C)NC(C3CC34CCCC4)=O)C2)=O)cc(F)cc(Cl)c1 c1(CC(C)C)oncc1C(=O)N(CCCNC(C1CC(O)C1)=O)CCO c1(C(C(=O)NC(C)C(=O)OC)N(C2CCCNC2=O)CC)ccc(F)c(OC)n1 c1(C(=O)NCC(C)(C2CCC2)NC(CC=C)=O)nc(Br)c2ccccn12 C1(NC(C=NOC)=O)CCCCN(C(C23CC(C)(C2)OC3C)=O)C1 c1(CNCC2(COC)C=CCN2)cccnc1O N1(C(c2cccc(CF)c2)=O)CCN(C(c2ccnc(O)c2)=O)C2CCCCC12 C1(C(N(CCCOCCNC(c2cc(C(N)=O)oc2)=O)C)=O)CC2CCCC2C1 Cc1nsc(C(N2CC(OCC(=O)NCC3(CO)CC=CC3)C2)=O)n1 CC1CC1C(=O)NCC(N1CCC1)=O.C12(CC1)CC(=O)N(C)C2 CN1CC(NC(c2ccc(CNC(=O)CC3CC4(CC4)CO3)o2)=O)C(F)(F)C1 Cc1ccc(C(N2CCC(CN(C)C(c3ccc(C4CCOC4)s3)=O)C2)=O)cc1 c1(OC)cccc2ccc(C(N3CCNCC3CC#N)=O)nc12.N12CCC1C2=O N1(C(C2C(CNC(C3C(OC(C)=O)C3)=O)CCC2)=O)CCc2nocc2C1 c1(C(=O)NCCC(C)NC(C2N(CC)CC2)=O)ccc(F)c2ccncc12 CC(C)CC(C)(CNC(C1(C#N)CCC1)=O)NC(c1nsnc1O)=O CCC(C)(C)CC(=O)NC(C(=O)NCC1CCCCN(C)C1)C(C)O C1(CC(=O)NC2CCN(CC)C2)CN(C(C2CCC(C)O2)=O)C(C)(C)C1 c1(C(=O)NCC2CN(C(=O)Cc3nc(Cl)cs3)CCO2)ccc2ccccc2n1 N1(C(C(CNC(C(C)c2cccs2)=O)CC2CC2)=O)CC(C)OCC1C c1(C(=O)NCCC(C)(C)NC(c2cnc(C(C)C)[nH]2)=O)ccc(Cl)c2occc12 CC1CNCCN1C(=O)C(=O)NCc1cccc(Cc2ccccc2)n1 C1(C(N2CC(C(F)(F)F)(OC)C2)=O)C2CC(O)C(C2)N1CC1(O)CS(=O)(=O)C1 CC(CCNC(=O)CC1(CO)CC1)NC(=O)CCN(S(C)(=O)=O)C Cc1nc(C)c(C(=O)NC2(C)CC(C(N3CC(C)(C)C3)=O)C2)s1 C1(Cc2n(C3CCCN(C)C3)nc(-c3cc[nH]n3)n2)COC2(CCC2)C1 CCCCC(F)C(=O)N1CCC(NC(C2CC(C)(C)C2)=O)C(O)C1 c1(C(N(CC(C)NC(C=NOC)=O)C2CC2)=O)cc(S(=O)(=O)N(C)C)oc1C CCCC(C)(O)CC(=O)N1CCN(C(c2nc3cccnc3s2)=O)C(CF)C1 C1(N(C(Cc2n(C)cnc2)=O)CCF)CCCN(C(=O)CSc2ccccn2)C1 C1(C(N2CCCC(N(C(=O)CCN3CCCC3)CC)C2)=O)CCn2nnnc2C1 c1(C(N2CC(O)CC(NC(c3n[nH]c(=N)s3)=O)C2)=O)ccc2oc(=O)oc2c1 N1(C(COC(C)=O)=O)CCC2CC2(C(=O)NCc2noc(C(C)C)n2)CC1 C(C)(C(C)C(=O)N1CC(CN2CCOCC2)C1)NC(c1cc(SC)on1)=O N1(C(Cc2c(F)ccc(N)c2)=O)CCC(NC(C23CCC2CC3)=O)C(CO)CC1 C(=O)(C1CCCc2[nH]nc(I)c21)Nc1cc(C)c(Br)cc1 CC(CCCCNC(=O)CN1CC(=O)NC1=O)NC(=O)Cc1ccco1 c1(C(N(C(CNC(CCCC(=C)C)=O)C)C)=O)[nH]nc2c1CCC2(C)C C1(CN(C(=O)C(c2cnn(C)c2)O)C)CC(F)CN1C(=O)Cc1cc[nH]c(=N)c1 C1(C(=O)NCC23C(CN(C(c4nn(C)c(C(F)F)c4)=O)C2)C3)CCCC12CCC2 C12(C(=O)NCCNC(c3nccnc3-n3ccnc3)=O)CCCCC1CCC2 N1(C(C(C)c2cc[nH]n2)=O)CC(NC(C2CC(F)(F)C2)=O)C(O)C1 N1(CC(=O)NCCCC(=O)NC2C(C)CCN(C(N)=O)C2)C(=O)C(=O)N(C)C1=O c1(-c2nc(-c3sc(C)c(Br)c3)no2)ccc([N+](=O)[O-])cc1 c1(OC)ccc(Cl)cc1CC(N1CCC(NC(=O)C=Cc2ccco2)C1)=O c1(C(=O)NCC(C)(CO)NC(Cc2c(CC)n[nH]c2CC)=O)cnc(O)c(C)c1 Cc1c(C(N2C3CCC2CN(C(c2ccon2)=O)C3)=O)nc2sccn12 C1(CN(C(c2c(C)c[nH]c2)=O)C)CCCCN1C(c1coc(C2CCCC2)n1)=O N1(C(CSc2nc(C)[nH]n2)=O)CCC(CC(C)NC(=O)Cc2cscn2)CC1 C1(NC(c2c(C)cno2)=O)CC(CNC(c2cnoc2C)=O)C12CCC2 c1(C(C(=O)NCCCOCCO)NC(CN(C)CC2CCCO2)=O)cnn(C)c1 N1(C(C(CCCOC)C)=O)CC2(C1)SCCC2NC(=O)C=Cc1sccc1C C(N=c1[nH]c2c(c(=NCCCn3nccn3)[nH]1)CCCCC2)c1c(C)ncs1 c1(CN2CC(CC(=O)Nc3cnc4cc[nH]c4c3)C2)cc(F)c(I)c(F)c1 c1(C(=O)NCCN(C(COCC=C)=O)C)ccc2c(Br)cnn2c1 CCC(C(=O)NCC12CC(CN1C(c1ccc(N(C)C)cc1)=O)C2)C(C)O C1(NC(=O)CCc2cncs2)CCN(C(C2CCS(=O)(=O)CC2)=O)C12CCCC2 C1(C(N2CC3CN(C(C4(C)CCC4)=O)CC3C2)=O)CC(c2ccc(F)cc2)=NO1 C=C(CNC(c1cc(C(C)(C)C)c[nH]1)=O)CCNC(c1cc(C(=O)OC)no1)=O c1(C(=O)OC)sc(Cl)cc1NCCCCC1CN(CC(F)(F)F)C1 c1(C(=O)NC23CC(NC(C4CCC5(CC4)CC5)=O)(C2)C3)noc2c1CCCCC2 C(=O)(C(F)(F)c1csc(Cl)n1)NC(c1cn(CCO)nn1)CCC Cc1cc2c(C(=O)NCC(CO)NC(=O)CSc3cccs3)cccc2[nH]1 C1(NC(=O)CN2CCOCC2)CCS(=O)(=O)C2(C1)CC(CNC(C1CCO1)=O)C2 CC12CC(CO)(C1)C1(CN(C(=O)C(c3cccc(F)c3)N3CCCCC3)C1)O2 CC(C)(C)CC(C)(C)C(=O)N1CCC2C(C(=O)NCC3(Cl)CC3(F)F)C2C1 CC1(CNC(c2ccc(CO)s2)=O)COCCN(C(c2coc3c2COC3)=O)C1 CCCCCCC(=O)NCCOC1CCN(C(=O)CCc2cccnc2)C1 C1(NC(c2ccon2)=O)CC2CC1N(C(=O)C=Cc1sccc1Br)C2 C1(O)(CNC(C(Cc2ccco2)NC(CC(C)OC)=O)=O)CCC(C)CC1 C1(C)(CNC(c2ccc(CC)c(F)c2)=O)CN(C(C2CC(CF)C2)=O)C(C)(C)C1 c1(COC(c2c(C(=O)OC)c[nH]n2)=O)cc(-c2ccccc2)cc(N)c1 N1(C(C(F)OC)=O)CCN(C(c2cc3n(n2)CCC3)=O)C(C(F)F)C1 c1(CC)ccc(F)cc1C(=O)NC(CNC(c1cccnn1)=O)C1CCC1 C1(C)(C(=O)NCCOCCCNC(C(CC)C)=O)CCN(C(C)=O)C1 C1(N(C(=O)CSc2nc[nH]n2)C)CN(C(c2ncncc2Cl)=O)CC1O N1(C(c2nc(C)oc2)=O)CC2C(CNC(=O)C(C)c3ccsc3)C2C1 c1(-c2nc(CC3(C(=O)OCC)CC3)on2)cc(C2CCC2)[nH]c1C C1(CNC(CCCC#N)=O)CCCCN(C(C2(n3cncn3)CC2)=O)C1 CC1CN(C(C2CC(CNC(=O)CC3CCC(=O)N3)C2)=O)CCO1 c1(C(N2CCCC(CNC(C=C(C)C(C)C)=O)C2)=O)ccc(Br)nc1N c1(C(N(C(C)C)CCNC(=O)C(O)C2CCCC2)=O)ccc(CN2CCCC2)cc1 c1(OCCC)cc(CNC(=O)NCC(c2ccc(C)nc2)CC)ccn1 CCCC(CC)CCC(=O)N1CC(=O)CC1C(N1CCCNC(=O)CC1)=O Cc1ccc(Cl)cc1C(C)NC(=O)C(C)(C)NS(N)(=O)=O c1(CC)ccc(N)c(C(=O)NC(C)(C)CN(C(=O)Cc2cc(C)sc2C)C)c1 C1(CC(=O)N(C)CC2N(C(Cc3ccc(OC)s3)=O)CCC2)C(=O)N(C)N=C1C C(CC(C)C(=O)N1CC2CC2(CNC(c2ccc(OCCF)cn2)=O)C1)OC S(=O)(=O)(c1ccc(Br)cc1NCc1cn(C)nc1Br)N1CCCC(C)(N(C)C)C1 CCC(CC(=O)N1CCC(CCO)CC1)NC(=O)COc1cccnc1C C(=O)(CC(C)C(C)(C)C)N1CCC(C(=O)NCc2nc[nH]n2)(CC)C1 C(C)(CO)(C(=O)NCC=C1CCN(C(C2C(F)(F)C23CC3)=O)CC1)OC c1(C(C(=O)NCCCCCNC(C(C2CCC2)OC)=O)(F)F)cccc(Cl)c1 c1(OC)ccc2c(n1)NC(C(N1C3CCC1(CNC(=O)C(C)(C)OC)CC3)=O)C2 C(=O)(NNc1ccc(NC)cc1Cl)NCCc1ccc(OC)c(C)c1 N1(C(C(COC)N(C)C)=O)CCOCCC1C(=O)Nc1ccc(O)nc1 C1(NC(c2cncnc2)=O)CN(C(c2ccc(CO)cc2)=O)CCC12CCC2 CC1CN(C(=O)CCc2ccccc2Br)CCCN1C(c1cccnc1O)=O CCCCCC(C)(C)C(=O)NCC1(NC(=O)CCn2[nH]c(=O)[nH]c2=O)CC1 c1(CN(CCNC(c2ccc(C3CCCCC3)s2)=O)CC)nnc(C)n1C C1(Nc2cc3nncn3cn2)CN(C(C2CC(N=[N+]=[N-])C2)=O)CC2(CCC2)C1 c1(C(=O)NC(COCC)C(=O)NC2CC2(C)C(F)F)cnn(C)c1Cl Cc1cnnc(O)c1C(N(C(CNC(=O)C=Cc1cn[nH]c1)C1CC1)C)=O N1(CCC)C(=O)NCC(N2CCC(n3ccnn3)C2)C1=O C(c1ccsc1C(F)(F)F)=CC(=O)OCC(C1CCS(=O)(=O)C1)=O CN1CC(C)(C(=O)NC2CC(O)CC2Nc2cc(F)ncn2)CC1=O c1(CN2C(C(=O)OCc3ncc(OCC)cn3)CC3CC32)c[nH]c2c(F)cccc12 O=C(NNC(=O)C1CCOCC1)C1CC(c2ccccc2)CN1 C(=O)(C(CCCS(C)(=O)=O)N(C)C)NC1CCN(C(c2c(C)n[nH]c2C)=O)CC1 Cc1ncc(C#N)cc1NC(C1CCCCCCN1C(=O)CC1CC1(C)C)=O C1(C(=O)Nc2c(C)ncnc2)CN(C(=O)CC2=CCCCC2)CC(C)(C)C1 c1(OC(C)C)ccc2c(C(=O)NCC3COC(C)(C)O3)ccnc2c1 N1(C(Cc2scc(C)c2)=O)CC2(C1)C(NC(C1C=CCCC1)=O)CCS2(=O)=O C1(CCOC)CN(C(C2COCCC2(F)F)=O)CCN1C(=O)C(F)=C1CCCC1 c1(CNc2c(C(=O)NC(C)=O)cccn2)c(C)nc(-c2ncccn2)nc1C.C1CC1 C(=O)(CCCCC(C)C)NCCOC(C)=O.c12ccc(C)c(c1)C(=O)N2 C1(NC(c2scc(C)c2)=O)CCC2(CCN(C(c3ccc(C#N)o3)=O)CC2)C1 C1(NC(=O)CC2=CCCC2)C2COCC1CN(C(=O)C(F)F)C2 CC12CCCC1N(C(c1ccc3c(c1)CCC3)C(=O)Nc1ccccc1Cl)CCC2 S(=O)(=O)(c1ccc(=NCCCCn2cnnc2)[nH]c1)NCc1cnn(CC)c1C c1(C(N2CCC(O)C2)=O)cc(Br)cn(COC2CC(Sc3ccc(C)cc3)C2)c1=O C(=O)(C(F)(F)C(F)(F)F)N1CC(CN(C(C(C(C)C)OC)=O)C)OCC1 C1(C(=O)NCC(c2ccccc2Br)N)CCC2(CCNCC2)C1 C1(NC(c2c(CCC)nns2)=O)CCN(C(=O)C2=NNC(=O)C2)CC12CCC2 c1(NC(C2C3(CN(C(CCn4c(C)cc(C)n4)=O)C3)C2)=O)cc(F)cc(F)c1C c1(C(N2CCC(C)(CNC(c3c(C)ccnn3)=O)CC2)=O)cccn2cnnc12 C(=O)(C1=CCCOC1)N1CCN(CCN(C)C(C2(F)CC=CC2)=O)CC1 C#Cc1ccnc(C(=O)NCc2ccc(CNC(C3CN(C)C3)=O)cc2)c1 CC(C(=O)N(C1CCCCC1)CC(=O)NC1CNC(=O)O1)S(C)(=O)=O C(=O)(C1=NOC(C)(C)C1)NC(C1CN(C(CCc2cccc(C)c2)=O)C1)C C1(C(=O)NCC2(NC(C3C(C)CC3)=O)CC2)CCC(C)(O)CC1 C=C=C(C)CC(=O)NC(C(C)SC)C(=O)Nc1ccc(CCF)cc1 CCN=C(NCC(C1CCCCCC1)OC)NCC(Cc1ccccc1)N(C)C C1(C2CC(=C)C2)NC(=S)N(CCCNC(=O)OC)C2=C1C(=O)NC21CCCC1 N1(C(c2c(CNC(C3(C(C)=O)CC3)=O)noc2)=O)CCCC2CC12 c1(OC(C)C)ccc(CC(N2CCCC2CN(C(=O)C(C)O)C)=O)cc1 C1(NC(CCCc2onc(C)n2)=O)CCCN(C(=O)C=CC2CCOCC2)C1 c1(SCC(N2CCOCC2)C(c2ccc(Br)cc2)=O)ccc([N+](=O)[O-])o1 C1(CNC(c2cc(OC)no2)=O)CCN(C(=O)Cc2ncc(Cl)s2)CC1O C(=O)(Nn1cnnc1C)C1C(NC(CCCOC)=O)CCCC1 c1(CN(C(N2CCCC2Cn2cc(C)cn2)=O)CC)ccc(O)cc1 c1(C(=O)NCC2CCN(C(C=C(C)C(F)F)=O)C2)ccc([N+](=O)[O-])cc1F CC1Cc2ccsc2CN1C(=O)Nc1ccc(C(=O)N=c2cc[nH][nH]2)c2[nH]ccc12 CCCC(C)(CC)C(=O)NCCC1CN(C(c2ccc(OC)o2)=O)CCO1 N1(C(C2CCC(CC)CC2)=O)CCC(NC(c2ncc[nH]c2=O)=O)CC(O)C1 C(C)(CCC(=O)N1CC2CC2(CNC(=O)C(C)(O)COC)C1)OCC C1(CC(=O)NCCCCCCNC(C)=O)CC(C)(C)OC1=O.C12CN(C1)C(C)(C)C2 C1(NC(=O)Cn2cc(C(N)=O)nn2)CCCN(c2ncncc2I)CC1 C1(NC(CC23CC(C)(OC2)C3)=O)CCCN(C(=O)CC2(O)COC(C)(C)C2)CC1 N1(C(c2cc(C)c(O)cc2)=O)CC(CNC(C2CC3(CCC3)C2)=O)N2CCC1C2 C(=O)(CC(C)(C)C(=O)OCC)N1CCC(NC(COCCCCC)=O)C(C)C1 N1(C(C2(C)CCCCO2)=O)CC2CCCC(C1)N2C(C12CCCCC1C2)=O c1(C(=O)OCC)cn2c(n1)CN(C(C)=O)CC2.c12cc(C#N)c(nc1O)[nH]2 Cc1cc(C(=O)N(C2CCCC(NC(=O)CSC(F)F)C2)C)ccc1C#N Cn1ncc(C(N2CCC(C(=O)NCC3CC4CCC3O4)CC2)=O)c1Cl c1(C(C(=O)N(CC(C)CNC(C2(CCF)CC2)=O)C)O)ccccc1F CCC(C)C(=O)C(=O)N1CCC(O)C(N(C(=O)C(C)NC(C)(C)CC)C)C1 c1(C(=O)NC(C(C)NC(=O)CCc2nnnn2C)C)c[nH]c2ccccc2c1=O c1(NCC(=O)NCC2(F)CC(NC(c3c(C)cccn3)=O)C2)ccccc1C#N Cc1cc(C(N2CC(CN(CC(O)COc3ccc(Br)cc3)C)C2)=O)cc(C)n1 Cc1n[nH]c(C)c1C(=O)NC1CCC1NC(=O)C=C1CCCCC1 N1(NC(=O)OC(C)(C)C)CCC(C(=O)O)C(CO)C1.c1(CC=O)noc(C2CC2)n1 c1(CC)cccc2c(CCNC(=O)C(C3CCC3)OCC)c[nH]c12 C#CCCN=C(NCc1ccc(Cl)c(F)c1F)NC1CSCC1C.CC(F)F C1(CC)C(C(N2CCC2)=O)CCCN1C(c1c[nH]c(C(N)=O)c1)=O c1(OC(F)(F)F)ncc[nH]c1=NCCc1ccc(F)cc1F c1(C2CC2F)cc(F)ccc1F.C1(=O)CN(S(C)(=O)=O)CCOCCN1C.C(=O)OC CCS(=O)(=O)c1ccc(C(=O)NCCCNC(c2cc(C(F)F)ccn2)=O)cc1 CN=c1nc(N2CCC(N(CC(C)C)C)CC2)[nH]c(=NCCP(C)(C)=O)[nH]1 N1(C(=O)OC)CCN(C(=O)C(F)n2cccn2)CC1.C12CN(CC1F)CC(=O)N2 N1(C(C2(C(C)NC(C3C(CC)OCC3)=O)CC2)=O)CCC2(CCCCO2)C1 N1(C(=O)C=CC(F)(F)F)CCn2ncc(CNC(=O)CCc3ccncc3)c2C1 C1(C(N2C(C)CCC2C)=O)CC2(CCCN(CC(c3ccc(Cl)nc3Cl)=O)C2)C1 c1(C(=O)NC(C(C)C)CCNC(=O)CC2CC3(CCC3)C2)csc(S(N)(=O)=O)c1 c1(CCC)nnsc1C(=O)NCC1(SC)CN(C(=O)C(C)CSC)C1 C(C)(C(C(=O)NCC(=O)N)C(C)C)NC(=O)OC.C12CCC(CC1)C(=O)NC2.C(CO)O c1(C(N(C(C)CNC(C2CC2C2CCC2)=O)C)=O)ccc2c(c1)nc(O)n2C C1(NC(C(CC)CC)=O)CCC2(CCCN(C(C3CCSCC3)=O)C2)C1 CC1OC2CCC1(C(=O)OCC(C)NCc1cccc(Br)c1)C2 C(C(=O)NC1(C)CC(C(=O)NCc2nc(C)c(C)s2)C1)(C(C)C)NC(C)=O CC(C)C(CO)C(=O)NC(C1CCN(C(=O)Cn2cc(Br)c(=N)[nH]2)C1)C C=C(C)CC(C(=O)N1CCCN(C(N)=O)CC1)NC(=O)C(C)c1ccco1 c1(NC(c2cn(C(C)C)nc2)C)cc(S(=O)(=O)N(CCCO)CC)ccc1C#N CN1CCN(Cc2ccc(-c3cccc(Cl)c3Cl)o2)c2ccc(Cl)cc21 Cc1cc(F)ccc1NC(C1COCC1NC(=O)CCNC(=O)CO)=O N1(C(C2CC(C)N(C)CC2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC12CCC2 C(=O)(CCC(C)NC(=O)C(O)CC1CCCC1)NCCCC(C)C N1(C(c2ccc(CC)cn2)=O)CC2CC(C(N3CC(N4CCOCC4)C3)=O)(C2)C1 C1(CC)(NC(=O)C(C)S(C)(=O)=O)CCCN(C(c2cn(C)cn2)=O)C1 C(=O)(C1CCCc2nnn(C)c21)NCCC(C)N(C(=O)CNC(N)=O)C c1(NC(C(n2cc(-c3ccccn3)nn2)C)=O)cccc(F)c1N S(=O)(=O)(c1cccnc1N1CCCC2(CCCO2)C1)NCC(CC)OC C1(C(N2CC(CC(=O)NC(C#C)CCC)(OC)C2)=O)OCCCC1(C)C C1(C2CCN(C(=O)CC3CCC(C)CC3)C2)(NC(c2c(C)ccc(Cl)c2)=O)CC1 C1(C(=O)NCC(C(=O)NCc2cc(C)ncc2)C)Cc2nccn2C1 N1(C(c2cn(CCOC)nc2)=O)CC(C2CCN(C(C3CCC(F)C3)=O)CC2)C1 N1(C(C2(C)CCC(C)C2)=O)CCC(CO)(CNC(c2[nH]nnc2C(F)F)=O)CC1 N1(C(C(C)OCCOC)=O)CCCN(C(C2(C#N)CC(F)(F)C2)=O)CC1 C1(CC)C(C(=O)NCCC2(O)CCC2)CCN1C(c1ccc(SC)o1)=O c1(C(=O)NC2C(C)(C)C2CNC(C2CC(C3CC3)C2)=O)ccccc1C1CC1 N(C1CCCCc2cnn(C)c21)C(C1N(C)CCN(C(=O)OC(C)(C)C)C1)=O c1(C(=O)NCC2CC=CCN2C(=O)CC2CCCO2)cnc(C(F)(F)F)c(F)c1 c1(CNC(CCCN(C(C(CC)OCC)=O)C)=O)cc(OC)ccc1C C(=O)(C(CNC(=O)C=Cc1cncn1C)C(C)(C)C)Nc1ccc(OC)c(O)c1 N1(C(=O)CCC2CCCOC2)CCC(O)(CNC(C2(O)CCOC2)=O)CC1 CN=c1[nH]c(-c2ccc(Br)cc2)c(CC(=O)OCCC2CCC(=O)NC2)s1 CC1CN(C(=O)CCCCc2cccc(O)c2)CC1NC(=O)C(=O)NCC1CC1 CC1CC2CCCCC2N1C(c1ccc2cc[nH]c2c1)C(=O)NC1(C)CC1 Cc1ccccc1-c1ccc(C(=O)NC(C)C(C)NC(C2CC(O)C2)=O)cc1 N1(C(c2c(CC)cc[nH]2)=O)CCC2C(CCCN2C(=O)CN2CCSCC2)C1 C1(NC(c2c(CC)nccn2)=O)(CNC(c2ncccc2Cl)=O)CC2CCC1C2 C(=O)(CC(C)C(=O)NC1CCCC(CC(=O)NCC(C)SC)C1)OCC c1(OC)nn(C)cc1C(N1CC=CC1C(=O)NCc1c(C)cnn1C)=O c1(C(N2C(CC(C)C)CC2)=O)coc(CNC(C2CCC(O)C2)=O)n1 C1(NC(C2CCCC2)=O)C2CC3CN(C(c4cnn5ncccc45)=O)C1C3C2 N1(C(c2c(C)cc(SC)s2)=O)CC(F)(F)CC1(C)CNC(=O)CCn1cccn1 C(=O)(CC(C(F)F)NC(=O)CCC1CCCN1C)N(C(C=C)C)C CC1CC(C(=O)NCC2COCCN(C(=O)CC=C(Cl)Cl)C2)=NO1 c1(C(=O)NC2C(NC(c3cc(C)oc3C)=O)C2)cnc(C(C)(C)C)nc1C CC1(C)CCC(C(=O)NC2(C)CCSCC2)(NC(C2CCC(C3CC3)C2)=O)C1 N1(SCC=CCOC(C2CC(CC)C2)=O)CCCCC1=O C12(CNC(CC3(C)CCCC3)=O)CN(C(=O)Cc3nc[nH]n3)CC1(C(F)(F)F)C2 C(=O)(C1CCCc2c(O)cccc21)N1CC(CCNC(C(C)OCCOC)=O)C1 c1(N(CCCNC(=O)Cc2ccsc2)CC)cc2nnc(C(C)(C)C)n2cn1 CC1CCC(NC(=O)CCP(C)(C)=O)CN1C(=O)CCOC(F)(F)F c12ccc(cc1)CN1CCN(CC1)C2=O.C1(CNC(CC)=O)(CF)CCC1 c1(C(N(C23C(C)OC(CC2)C3)C(C)C)=O)ccnc2c1ccn2C NC1C2CCC3C(C2)C13C(N1CCC(c2cc3cnccc3[nH]2)CC1)=O Cc1c(Cl)nc[nH]c1=NCC1(CNC(=O)CC2(C)CC2(F)Cl)CC1 N1(C(c2c(=N)[nH]cnc2)=O)CC2CC(C(=O)NCCC3(CO)CC3)CC2C1 c1(CNC(=O)NC)ccc(O)cn1.C=C(Cl)CN C12(C(=O)OC)CC(NC(=NC)NCC3CCCC3N3CCCC3)(C1)C2 CC1CCC2(NC(=O)N(c3ccc(CC#N)cc3)C2)N(CCSC#N)C1 c1(C(=O)Oc2ccc(C3OCCN(CC)C3)cc2)ccc(S(=O)(=O)NC)s1.OC CC(CC(F)(F)F)N=c1[nH]c2c(c(=NC3CC(=O)N(CC(F)(F)F)C3)[nH]1)CSC2 C1(CC(=O)NCC(C)NC(C2CCC(SCC)CC2)=O)CCCC2(CCC2)O1 C1(NC(CCC#CC)=O)CN(C(c2cc3sccc3s2)=O)CCC1C c1(C(N2CCN(C(C(C)C#N)=O)CC2)=O)nc(C(F)(F)F)n2ccncc12 c1(C(=O)Nc2c(C)cccc2O)cc2c(Br)coc2cn1 CCCC(CC)CC(=O)NCCCC(C)(C)NC(c1ccnc(Cl)c1N)=O Cc1cc(=NCc2ccc(C(F)F)nc2)[nH]c(N(CC(C2CCCCC2)C)C)n1 c1(C(=O)NC2CN(c3ncc(C#C)cn3)C(C)CC2)cc2c(C)ccc(F)c2o1 c1(C(=O)Nc2cccc(CNC(CC3CCCC(C)C3)=O)c2)nnc2ccccn12 C1(C(N2CCN(C(C(C)(C)n3ccnn3)=O)CC2)=O)CCC2CC1CO2 C1(C)(C(N2CC(CN(C(c3cc(CC)on3)=O)C)OCC2)=O)CCCNS1(=O)=O c1(NC(c2c(CC)cccc2)C(=O)Nc2ccccc2CO)ccc(C)c(F)c1 c1(N2CC(O)CC(OC)C2)cc(S(=O)(=O)N(C)CCF)ccc1C#N C(c1cccc(F)c1)=C(C(=O)N(CC(CNC(Cc1nnc(C)n1C)=O)C)C)F C(=O)(C1=C(Cl)CCC1)N1C(CC)C(C(=O)Nc2cn(C)nc2C)CC1 N1(C(COc2n(C)ccn2)=O)CCN(C(C2CC2CF)=O)C(c2ccccn2)C1 c1(C(N2CC(NC(C(CC)OCC)=O)C2)=O)ccc2cc[nH]c2n1 c1(C(=O)NCC2(F)CCN(C(C3CCCS3)=O)C2)ncn2ccccc12 C(CCN(C(=O)C(N1CCSCC1)C)C)(C(C)C)NC(Cc1nc(C)[nH]n1)=O C1(C(N2CCCCC(NC(C(C)OC)=O)C2)=O)CSC(c2ccccc2)=N1 C(=O)(C1CCCc2c1ncn2C)N1CCCC(CNC(C(C)OC2COC2)=O)C1 C1(C)(C(N(CCOC)CCNC(=O)CC2(C(F)(F)F)CC2)=O)CCCC1CC c1(C(=O)NCCCC(C)(C)NC(C2CC2(F)Cl)=O)ccc2ncnn2c1 CCCC(C(O)C(=O)NCC(C)(C)CN(C)C)NC(=O)C(C)(C)CCOC C1(NC(=O)C=CCO)CS(=O)(=O)CC1NC(c1cscc1Br)=O C1(CNC(C(C)N(C(C2CCC3(CCC3)C2)=O)C2CC2)=O)OCCCC1(C)C c1(C(N(CCNC(c2cc(OC)ncc2)=O)C2CC2)=O)c(C)ccc(Cl)c1F C1(N(C(C=NOC)=O)C)CN(C(=O)C(C)(C)c2ccc(Cl)s2)CC1F N1(C(c2cnc(C)o2)=O)CCC(NC(c2c(Cl)nsc2Cl)=O)CC(C)(C)C1 Cc1ccc(C)c(C(=O)NCC2C(C)CCN2C(c2cccc(C)c2C)=O)c1 c1(CC)ccc(NC(=O)CCOc2ccccc2OCC(=O)NC)c(C)n1 N1(C(c2c(C)ccnc2)=O)C2CCC(C2)C1C(N1CCCC1c1ncc[nH]1)=O c1(C(C)(C)C)n[nH]cc1C(=O)NC1CCCC1NC(=O)C(F)C1CN(C2COC2)C1 c1(CN2CC(C(=O)Nc3c(C)ccc(Br)n3)SCC2)nc2ccccc2s1 c1(CC#N)cccc(C(N2CC(O)CC2C(=O)NCC2CCC(=O)O2)=O)c1 C1(CNC(C2CC(NC(C(=Cc3ccco3)C)=O)C2)=O)CC(O)C(O)C1 c1(OC(C)C)cccc(CN2CCC(CO)(NC(C3CCC3)=O)C2)c1F C1(C2CCCN(C(c3cc(F)c(C#N)c(F)c3)=O)C2)(NC(CNC(C)=O)=O)CC1 C1(NC(CCc2cncc(C)c2)=O)CCCC(N=c2nc(Cl)[nH]c(C)c2C#N)C1 C1(CNC(c2n(CC)ccn2)=O)CC2(CO1)CN(C(C1CCSCC1)=O)C2 CC(C)(C)CC(O)C(=O)NC1CN(C(=O)C=Cc2ccc(Cl)s2)CC2(CC2)C1 c1(CSCC(=O)NC(C(c2ccccc2Cl)OC)C)ncc2c(n1)CCCCC2 N1(C(CNS(N)(=O)=O)=O)CC(O)(C2CCN(C(C3(c4cccnc4)CC3)=O)CC2)C1 N1(C(CC2(C)N(C(c3cc(CC)ncc3)=O)CC2)=O)CCC(OC)C(C)(C)C1 C1(NC(c2cnn(CCNC(=O)C(O)C3CCCC3)c2)=O)CCCCCC1O C1(CNC(C2(C(C)C)CC2)=O)CCC2(CN(C(=O)CCn3cccc3)C2)O1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCOC)CCNC(=O)CC1CCCC(=O)C1 C1(NC(CC2(N(C(c3c(C)cn(C)c3)=O)C)CC2)=O)CCOC2(CCC2)C1 C(=O)(C(F)(F)CC(=O)NCC(CNC(c1cc(OC)ncn1)=O)OC)OC c1(N(C2CCN(C(C3CC3(C)C)=O)C2)C)ncnc2c1ncn2C(CO)CO C1(C(=O)NCC(CNC(C(C2CC(C)(C)C2)OC)=O)(C)C)CCCS1(=O)=O C(=O)(C(O)P(C)(C)=O)NC1CC(NC(C(COC)(C)OC)=O)C1 C12(CNC(CC(=O)N(C)C)=O)CC3CC(CC(NC(C4CCOC4)=O)(C3)C1)C2 C1(N(C)C(c2cncc(F)c2)=O)CCCCN(C(C2CC(CF)C2)=O)C1 CCCC(CCC)C(=O)NC1C=CCN(C(=O)Cc2nncn2C(C)C)C1 C(C)(CC(=O)N(CC(C)(C)NC(C1CC12CC2)=O)C)SC Cc1nnc2cc(C(N3CCc4c(Br)ccnc4C3)=O)ncn12 N1(CC(=O)NC(CNC(C2CCC(C(=O)OC)C2)=O)(C)CO)CCCCCC1=O c1(OC(C(=O)NC(CC)CNC(c2cccc(Cl)c2)=O)(C)C)cccc(C)c1F N1(C(C(C(C)C)SC)=O)CCC(C2(O)CN(C(=O)C(C(C)C)SC)C2)CC1 CC1CC(CCNC(c2ccnnc2)=O)CCN1C(c1cc(C2CC2)no1)=O c1(CCN2CCCC(NC)C2)ccc2c(c1)[nH]c(=O)[nH]2.C(C)(C)(C)O.CN c1(OCC)ccc(Cl)c(C(N2CCC(NC(=O)COCCSC3CC3)CC2)=O)n1 O=C1CC(C(=O)NCC=CC(=O)NC2CC(CC(F)(F)F)C2)NC(=O)N1 C1(C(=O)NC2(C)CC(NC(c3c(CCC)occ3)=O)C2)CC(=O)N(C)C1 C1(CC)CN(C(c2ccc(F)cc2OC)=O)CCN1Cc1ccc(C(C)C)cc1 N(C(=NCC1C=CCCC1)NCC1(C(F)(F)F)CCCC1)C(CC)C c1(C(N2C(C)C(NC(C3CCC4(CCC4)O3)=O)CC2)=O)cc2n(n1)CCN(C)C2 CCCC(CCCNC(=O)C(C)(C)C1CCOCC1)NC(C1CC(C)C1)=O CC(C(C)(C)NC(c1cc(F)c[nH]1)=O)NC(c1cncn1C)=O C(=O)(N=c1ccn(C(C)C)[nH]1)c1cc(CNC(CC2ON=C(C)C2)=O)[nH]n1 Cc1ccc(C(=O)N(C2CCN(CCCN3CCCC3=O)CC2)C)cc1Cl C1(CN(C(=O)CCOCC2CC2)C)CCCCN1C(=O)CC1CCC1(F)F C1(CNC(c2cc(CO)[nH]n2)=O)CN(C(C2(CF)CCOCC2)=O)CC1(F)F C1(N(C)CC)CCCN(C(=O)C(C(C)C)NC(=O)NC(C)C)C1 c1(-c2onc(C(C(C)C)OC)n2)cccc(OC(C)C(=O)N(C)C)c1 CCCC(CC(C)C)C(=O)NC1CN(Cc2ccsc2)CC1(C)C c1(C(=O)NCC(CN(C(=O)Cc2ccnn2C)CC)(C)C)nc(Cl)ccc1N N1(C(C2CCN(CC)CC2)=O)CCC2OCCN(C(=O)Cn3cc(C)cn3)C2C1 N1(C(CN(CC)NC(c2cc(C)sn2)=O)=O)CC(O)(CCc2ccccc2)C1 c1(OCCCC)ccc(C(=O)NCC(C)NC(C2C(C)C2(F)F)=O)cc1 Cc1ccc(F)cc1C(N1C(C(=O)NCCCN(C)C)CC(C)C1)=O.C(C)(C)(C)S Cc1ccn(CC(C)C(=O)NC2CC2CNC(=O)C=CCN2CCOCC2)n1 c1(C(=O)NCC(C(C)C)NC(C2CN3CCN2CC3)=O)cnc2ccccc2c1 N1(c2ccnc(C(=O)OC)n2)CC2CCC1CN2C(=O)CSCc1cccs1 C1(SC)CN(C(C2CC2C(=O)NCCO)=O)CC1NC(C1CCSCC1)=O c1(OC)cc(C(=O)NCC2CC2NC(C2CCCC2F)=O)ccc1OC(C)C C1(C(=O)NCCC2N(C(CC(C)N(C)C)=O)CCSC2)CCc2nncn2C1 C1(NC(c2c(N=[N+]=[N-])cccc2)=O)CCCCC12CCN(C(C1CC1(F)F)=O)C2 C(CCCCCS(N)(=O)=O)NC(=O)NC1ON=C(C(C)C)C1 NC1CCCC(CNC(=O)CCNCc2ccncc2C(F)(F)F)C1 C=C(C)CCCC(=O)NCC(C)C.C(C)(C)(CO)OCCNC(=O)C(C)OC C1(C(=O)NCC(CCOC)NC(c2ccco2)=O)CCC(=O)N(C2CC2)C1 N1(C(=O)C=CCF)CC2(CCN(C(=O)Cc3ccccc3)C2)C1 C1(NC(c2ccc(F)nc2)=O)COC2(C1)CN(C(c1nc3cccnc3s1)=O)C2 CCC(C)C(O)C(=O)N1CCSCC1CCNC(c1ccc(F)c(C)c1)=O C1(NC(c2ccc(CC(C)C)cc2)=O)C(C)CN(C(c2ccnn2C)=O)CC1C N1(C(C(C)=CC)=O)CCN(C(=O)CCc2cc(C)sc2C)CC1c1cccnc1 C1(NC(C2CC(CCC)C2)=O)CC(C)CN(C(c2cc3occc3[nH]2)=O)C1 C1(CC(=O)NC2CCN(C(=O)CCN3CCC(F)C3)CC2)(OC)CCCCC1 C1(NC(=O)COc2cccnc2Cl)CC2CCC1CC2NC(C1CC(O)C1)=O C1(C(N(CC(C)C#N)CC)=O)C2CC3C(C2NC(C2CCCC(CF)C2)=O)C13 N1(C(C(CC)N(CC)CC)=O)CCC2CC1CN(C(C1C3(CC3)C13CC3)=O)C2 c1(CNC(CN(C(C(C)OCC#C)=O)C)=O)ccc(O)c(F)c1 Cc1ccc(C2(C(N3CCCC(NC(C4CN(C)C(=O)N4)=O)C3)=O)CC2)cc1C CC(C(C)(C)NC1CC(C(=O)O)C1)C1CCCC1 C1(SC)C(=O)NOCC(=O)Oc2ccc1cc2.N1(C(C)C)CCCC1 C1(F)(C(N(C2CCN(C(C3(C(F)(F)F)CCCC3)=O)C2)CCC)=O)CCOCC1 C1(C(N2CCN(C(=O)CCC34CCC(CC3)C4)CC2)=O)CC12CCS(=O)(=O)CC2 CCC(CC)C(F)C(=O)N1CC(O)(CNC(=O)CC(C)C(=O)OC)C1 C(=O)(C(F)(F)CO)N(CC(CC)N)CC.CCCC(=O)NCC C1(C(=O)OCC(=O)C2CC2)CC(F)(F)CS1.Cc1noc(CN)n1.N1CC2(C1)CN2 c1(C(=O)NCCC2CN(C(COCCCC#C)=O)C2)c(C)nsc1NC1CC1 C1(C(C(=O)N2CC(N(C)C)C2)(C)C)CCN(C(=O)CCc2cnco2)CC1 C1(NC(C2(C)CC(C)C2)=O)CC2CC(NC(c3cncc(F)c3)=O)C1C2 CCCC(C)(C)CC(=O)NC(C)CN(C)C(c1ncc(F)cc1N)=O c1(SCC)cccc(C(=O)NCCC(C)N(C)C(c2sc(=N)[nH]c2C)=O)c1 C1(NC(C(C)C)=O)CC(C(=O)Nc2ncccc2C(C)C)CC1O N1(C(CC(CC(C)C)C)=O)CCCC2(C1)CN(C(c1cccc(C#N)c1)=O)C2 N(C1CCc2ccc(Cl)cc21)C(C1CCCN(CC2CCN(CCC)C2)CC1)=O c1(C(C(=O)NCCC2CCN(C(C(C)=CC)=O)C2)SC)ccc(Cl)cc1 c1(C(N(C)CC2N(C(C(C)OCCCCCC)=O)CCC2)=O)ccc(O)nn1 C1(NCCOC)C=CS(=O)(=O)C1.C(C)(C(=O)NCCON(CC)CC)NC(C)=O C1(C(=O)NC2C(NC(COC(CC)C)=O)CCCC2)CC(C)OC(C)C1 N1(C(c2ccc(S(=O)(=O)N(C)C)cc2)=O)CCC2OCCN(C(=O)CNC=O)C2C1 N1(C(CCSC)=O)CCCCC1C(=O)NC1CN(C(c2ccon2)=O)CC1O C(=O)(C1c2c[nH]nc2CN1C(c1ccc(C#N)s1)=O)NCCCN(C)C CCC(CCOC)C(=O)NC12CC(NC(C3(c4ccc(O)nc4)CC3)=O)(C1)C2.COC CC(C)CC(=O)N(CCC(=O)NCCCn1cc(CNC(C)(C)C)nn1)CCO C(=O)(C(F)(F)C=C)NC(C1CCN(C(=O)CCCCN2CCCC2)CC1)C C1(CNC(CCOC(C)=O)=O)CCN(C(C2CC(F)(c3ccccc3)C2)=O)C1 C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)CSC(F)F)CC12CCC2 c1(-c2cccc(C)c2)cc(C(=O)N(CC(C)C(C)C)C)ccc1OC(F)F N1(C(C2(C)CC(C)C2)=O)CCC2(CCCN(C(=O)CCS(C)(=O)=O)C2)C1 C12(C(=O)NCC3(OCC)CCOC3)CCCC1CC2 C=C(C)CN=C(NCC1CCC(C)O1)NCC(c1cc2ccccc2[nH]1)(C)C C1(C(=O)NC2C(CC)C2)CN(c2cc(C(=O)OC)ccn2)CCC1O N1(C(CC(C)(C)C)=O)CC2OCCN(C(c3cccc(Cl)c3F)=O)C2C1 c1(CNC(C(C)NC(c2cccnc2)C(=O)OCC)=O)nnc2ccccn12 c1(C(C)=O)cc(C)nc(N2CC(NC(C3CC4(CCC4)C3)=O)C(F)C2)n1 CCC(C(=O)NC1(CN(C2CC=CC2)C(c2ccccc2)=O)CC1)C(C)(C)CC N1(C(Cc2ccc(C)s2)=O)C2CCC1C(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 C(CCCC(=O)Nc1cccc(OCCN2CCN(C(=O)C(F)F)CC2)c1)OC c1(CN(C2CC3CNC2C3)C(C2CCC2)=O)ccc(C(F)(F)F)cc1 Cc1nn(C)cc1CC(=O)N(CC(C)CNC(c1ccncc1C(F)F)=O)C C12(CNC(C3CC(=C)C3)=O)CCC(C1)N(C(C1(N(C)C)CCCCC1)=O)C2 N1(C(Cc2cnc(C)o2)=O)CCC(C)C1CNC(C1CC(C)C1)=O c1(C(N2C(C(=O)Nc3cc(C)nc(Cl)c3)CC3(CC3)C2)=O)cn2cc(Cl)ccc2n1 C1(COC)CN(C(=O)CCC2CC2(Cl)Cl)CCN1C(c1cccn1C)=O C(=O)(CCC(C)(C)C(=O)N(CCCN(C)C(c1cccc(=O)n1C)=O)C)OC c1(C(=O)NCC(C)N(C)C(C2(C)CCCS2)=O)ccc2[nH]c(=N)n(C)c2c1 CC1=C(C(=O)NC2CN(C(c3nccc(Cl)c3F)=O)CC2C)CCC(C)(C)C1 N1(C(C(C)c2cccs2)=O)CCN(C(=O)CCC2CCC(=O)NC2)CC2(CC2)C1 c1(OCC)ccc(NC(=O)CC2CCN(C(=O)Cn3cc(CO)nn3)CC2)cn1 c1(C(N(C2CCC(NC(Cc3c(C)noc3)=O)C2)C)=O)cnc2[nH]cnc2c1 CCC(O)C(C)C(=O)N(C1CCN(C(c2cnc(OC)nc2C)=O)CC1)CCO C1(c2cccc(C)c2)CC(C(=O)NCC23CC4CC2C3C4O)=NO1 C(C(CO)C(F)(F)F)NC(C(c1cnn(C)c1)NC(c1cn(CC)nn1)=O)=O N1(C(c2c(C)cno2)=O)CC2CCC1C2NC(c1cc2n(n1)CCO2)=O N1(C(C(CCOC)C)=O)CCC2(CCCN2C(=O)CCSCC(C)C)CC1 c1(C(=O)NC(CN(C(c2cc(CCC)ncc2)=O)C)C)nc(C)ncc1Cl c1(C(N(CC(CC)NC(c2sccc2CO)=O)C)=O)cc(CO)on1 c1(NC(C(C2(O)CN(C(C(C3CC3)OC)=O)C2)F)=O)cnccc1CO CCC(CC)CCC(=O)NC(C(=O)NCCN(CCCF)C)C(C)C C(CCCC(=O)NC1(C(N2CCC(n3ccnc3)C2)=O)CCN(C)C1)SC c1(CC(=O)NCC(C2CCCCC2)NC(=O)Cc2c[nH]nc2O)ccccc1Cl c1(C(N2C(CNC(=O)C(F)n3ccnc3)COCC2)=O)ccc2c(c1)COCC2 C=CCC(C)(CC)C(=O)NC1CC(C)CN(C(c2cccc3nncn23)=O)C1 C(CNc1ccc(Cl)c(Cl)c1)(C(C)(C)C(C)C)NC(C)=O Cc1nc2c(s1)CCCC2C(=O)N1CCCC(C)(NC(=O)C=CC2CCOC2)C1 N1(C(c2c(CC)cccc2)=O)CC(NC(c2cc(C)ccc2F)=O)CC2(CC2)C1 N1(Cc2c(F)c(Br)ccc2)CCCc2oc(Br)cc2C1 c1(C(=O)NC2C(C)N(C(=O)CCc3cccc(O)c3)CC2)ccc(F)c(Cl)c1 C1(NC(C2(OC)CCOC2)=O)C2CC1N(C(c1cc(C3CC3)nn1C)=O)C2C c1(NCCCCCCSC)[nH]c(=NCc2cc(C3CC3)no2)nc2c1cnn2C C1(NC(C2C(C)C2)=O)CC2CCC(C1C)N2C(C1CC2CCCCN2C1)=O c1(C(N(CC(CNC(C(C)OCC#C)=O)C)C)=O)cc(C(C)C)on1 C1(C(C)NC(C2CN(CC(F)F)C2)=O)CCN(C(=O)Cc2cccc(O)c2)CC1 N1(C(C2(N(C)C)CC2)=O)CCCCC2(CCN(C(C3CCC(CO)CC3)=O)C2)C1 CC1=C(C)CC(C)(C(=O)NCC(C(C)C)NC(C2(C)CCCC2)=O)CC1 N1(C(C2=NOC(C)C2)=O)CCOCC12CCN(C(=O)CNc1nccs1)C2 C(CCCCC(=O)NC(CCN(C(=O)CC1CCCOC1)C)C(C)C)OC c1(C2(CC(=O)NC3C(CNC(=O)CCc4ncc[nH]4)C3)CC2)ccccc1 C1(CNC(c2c(OC)ccnc2F)=O)CCC2(CN(Cc3nc[nH]n3)C2)O1 c1(C(=O)NCC2(CC(=O)N(C)C)CCOCC2)ccc(F)c(O)c1 c1(C(=O)NCCN(C(=O)CN2CCC2C)C(C)C)ncc(Cl)cc1Cl N1(C(c2ncc(C)cc2C)=O)CCCCC1C1CCCN1C(=O)C#CC(C)(C)C C(=O)(C#CC1(C)CCCO1)NC(C(=O)NCC1ON=C(CC)C1)C1CCOC1 C1(C(N2C3CN(C(C(CCCC)=O)=O)CC2CC3)=O)C2Cc3cc(Cl)ccc3C12 N1(C(CC2CCC(NC(c3nsnc3O)=O)C2)=O)CCC2(C=CCO2)CC1 C(=O)(CCC(F)(F)F)NCC1CN(C(c2ccc(CC)[nH]2)=O)CC1C Cc1csc(CC(=O)NC2CC(F)(CNC(=O)C(C)CC3CCC3)C2)c1 N1(C(C(CC)O)=O)CCC2(CCCN(C(=O)Cc3ccc(C)cc3C)C2)C1 CCCCCCCC(=O)NCC1(NC(C2CN(C(C)=O)C2)=O)CCC(C)(C)CC1 C1(C(=O)NCCO)(CC)CCN(C(=O)CSCCC(C)C)C1.C1CCO1 c1(C(N(CC(CNC(C(C=CC)O)=O)C)C)=O)ccc(C(C)(F)F)nc1 CC1CCCCC1NC(=O)CC(c1ccccc1)N.N1CCCC1 N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCN(C(C23CC2C3)=O)CC1CO C(N=c1[nH]c(=NCc2nc3cnccc3[nH]2)c2ncccc2[nH]1)c1snc(C)n1 c1(C(=O)Nc2ccc(C)cc2)cc(Br)nc(Br)c1.C12CCCC1NC(=O)C2 C#CC1(C(=O)NC(C)CC(C)O)CN(C(=O)CCc2ccco2)C1 N1(C(c2c(OC)cc(C)s2)=O)CCC2(C1)CN(C(C13CC(C)(C1)C3)=O)C2 CC#CCC(C(=O)N(C1CCC(C)(C)CC1)C)NC(c1cn2c(n1)CCC2)=O N1(C(c2c(C)scc2)=O)CC2(C1)CN(C(C1(C3CCCCO3)CC1)=O)CCO2 C1(N(CCCCCCC=C)C)=CC2=NCCC(=N1)N2.N1CCC(OC)(OC)C1 C12(CNC(c3ncn(CC)c3)=O)CCC(CC1)N(C(c1cc(Cl)sc1Cl)=O)C2 Cn1ncc(CN2CCC(c3nnc(C(F)(F)F)s3)C2)c1F c1(CSCC)ccccc1C(=O)NCCCCNC(=O)CCC(=O)N(C)C Cc1onc(CO)c1C(=O)NCC(N1CCN(C(C2CCSCC2)=O)CC1)=O c1(C(=O)NCC(C)C(N2CCCC2(C)C2CC2)=O)cnc(=N)[nH]c1 C(C(O)CC(=O)N1CCCC(CCNC(c2cc(C(N)=O)cs2)=O)C1)N(C)C c1(C(=O)NC(c2noc(C3CC3c3ccccc3)n2)C2CC2)ccc(Cl)cn1 CCC(C(=O)NCCC1(NC(c2coc(CO)n2)=O)CCC1)C(C)C C1(NC(c2c(C(N)=O)coc2)=O)CN(C(c2cc(Br)ccn2)=O)CC1F c1(C(N2C(CC(=O)NC(C3CCCC3)CO)C=CC2)=O)cncc(Cl)c1 c1(C(N2CCOCC(CNC(CCOCC)=O)C2)=O)cc2ccc(OC)cc2[nH]1 C(=O)(CCC(C)(F)F)NC(C1(O)CN(C(C2CC2C2CC2C)=O)C1)C N1(CC(C)NC(=O)CC(C)(C)C)CCN(C(=O)CC(C)N(C)C)CC1 c1(C(=O)NCC(C)NC(COC2C(COC)CCCC2)=O)ccc(C)cc1C c1(OC)ccc(Cl)cc1C(N1CCC(NC(=O)C2=COCCO2)C(F)C1)=O N1(C(=O)C2CC2)CCOC(CN2CC(CC3CCCC3)C2)C1 C1(Nc2ncnc(=N)[nH]2)CCCC2CN(C(=O)Cc3csc(C(C)(C)C)n3)CC12 CCC(C)(C(=O)NC1CC(OC)CN(C(C2CCCN2C(C)=O)=O)C1)C(N)=O CCC(CC(F)F)C(=O)N1CCOCC1CNC(c1nn(CC)cc1Cl)=O N1(C(C2N(C(C3CCC(CC)OC3)=O)C3C(C2)C3)=O)CCC(O)(COC)CC1 CC(C)CC(CNC(c1cccnc1S)=O)C(=O)N1CC(c2ccncc2)C1 C1(CC(=O)NCC2(CN)CCC2)COC(=O)C1.C12(CCC1)CC(=O)N2 N1(C(C2(OC)CCOC2)=O)CC2(CCCC2NC(c2cccc(C(C)=O)c2)=O)C1 CC1(NCCc2ccsc2)CN(CC2CC(F)(F)C2)C1 c1(C(=O)NCCCCN(C(=O)CC(C)(C)O)C)cc2cc[nH]c2cn1 C1(C(=O)NC(C)C(C)F)(NC(c2c(C)occ2)=O)CCN(C)C1 c1(C(=O)NCC(CNC(c2c(C)scc2)=O)(C)F)ccc(N)c2ccncc12 c1(CN(C)C(c2cnncc2O)=O)ccc(CNC(C2(C)C=CCC2)=O)cc1 c1(C(=O)NC2(C)CCCC2)ccc(NCCNC(=O)CP(C)(C)=O)cn1 CC1CC2CN(C(C3COCCC3NC(C3CCC(CO)CC3)=O)=O)CC12 C1(CNC(CNC(C)=O)=O)CN(C(c2coc(Cc3ccccc3)c2)=O)CC1O c1(C(=O)NC2CC(NC(C3CCC(NC(C)=O)C3)=O)C2)ncccc1S(C)(=O)=O CCCC(CCNC(C1CC(NC(=O)Cc2csnn2)CCO1)=O)CCC C12(C(=O)NCCCCOC(C)C)CC(CN1C(C1CC=CCC1C)=O)C2 N1(C(C(CC)=O)=O)CC(NC(=O)OC(C)(C)C)CC1(CC)CC C(=O)(C1=CCCOCC1)NC1CCCC(CNC(C2C(C)C2)=O)C1 Cc1ccc(C(=O)N(C)CC=CC(=O)NC2CC(=O)N(O)C2)c(F)c1 C1(N(C(C(c2cncc(Cl)c2)OC)=O)C)CC(NCCSC)C12CCC2 c1(NCCOC)nc2ccccc2nc1NCCOC1CC1.c1(O)ccccc1C N1(C(Cc2nc(C)sc2)=O)CCCN(C(C2CC3(CCC3)C2)=O)CC1C c1(COCC(C)(C)C)nc(=N)cc[nH]1.C(CC(=O)NC1CC1)OCC=O C1(NC(C(CC)n2cncn2)=O)CCCC(NC(c2cn(C(C)C)nc2C)=O)C1 CCCCCC(C)(CC)C(=O)N(CCC)CCNC(c1csc(C(N)=O)n1)=O c1(C(=O)NC(C2CC(NC(C3OCCC3(C)C)=O)C2)C)ccc(O)cn1 S(=O)(=O)(c1cnn(-c2ccc(Cl)c(Cl)c2)c1)NC(C)CC1(O)CCCOC1 c1(C(=O)NCC(C)(O)CNC(=O)CCNC(=O)CO)ccc2cc[nH]c2n1 c1(CC(=O)N(CCN(C(C(c2ccccc2)C)=O)C)C)ccc(C2CC2)c(F)c1 C1(CNC(CC(C)F)=O)CC2CCCC2N1C(=O)Cn1cc(Br)cn1 C1(NC(CC2(NC(C)=O)CC2)=O)CCCC1NC(c1sccc1CN(C)C)=O C1(CNC(=O)COc2ccsn2)CCN(C(=O)CC2CCCS2(=O)=O)CC1(F)F C1(CNC(Cc2nc(C)c(C)[nH]2)=O)CC(C)CN(C(C2(CC(F)F)CCC2)=O)C1 N1(C(C=CC(C)(C)C)=O)CCC(NC(c2c[nH]nc2F)=O)C1 N1(C(c2c(C)nc(CC)o2)=O)CCC(NC(C2SCCS2)=O)C2(CCC2)C1 C(C(O)C(F)(F)C(F)(F)F)NC(C(=O)NCC1(C)CCOC1C1CC1)=O C1(NC(=O)Cc2cccs2)(CNC(c2cnc(C3CC3)s2)=O)CC2CCC1CC2 C12(CC(N3CC(NC(c4c(C)nn(CCO)c4)=O)C(F)C3)=O)CNC(=O)C(C1)C2 C1(CC(N2CCCCC2COCc2nn[nH]n2)=O)CCCCCC1(F)F C(=O)(CC1=CCCC1)NC(C(C)(C)NC(C1CCC(CC)CC1)=O)C C(=O)(CC1C(=O)Nc2ccccc21)NC1C(NC(C(C)OC(C)(C)C)=O)COC1 CC(CC(=O)N(C1(CC(N2CCC(C3CC3)CC2)=O)CC1)C)C(F)(F)F C(=O)(N=c1nc(Cl)nc2[nH][nH]cc1-2)C1N(C(c2ccc(C)cc2)=O)CCC1O CC1(C)CC(C)(C(=O)NC2C3CC(NC(c4ccon4)=O)CC23)C1 N1(C(CCNC(c2c[nH]nc2-c2ccncc2)=O)=O)CCC(C(C)OCC)CC1 C1(C(=O)N2CC(n3cc(C4(CO)CC4)nn3)CO2)CCC2C1C2(F)F C(=O)(CCCCCCNC(c1cnn2ccccc12)=O)NC(C1CCCOC1)C CC(C)C(CCN(C)C(C1CCC(F)(F)C1)=O)NC(C1(CCF)CC1)=O C1(CNC(CC2CCC(C)CO2)=O)CN(C(C2OCC2(C)C)=O)CCCO1 C1(NC(C2(C#N)CCCC2)=O)CC2CCC1N(C(=O)CCN1CCNC(=O)C1)C2 N1(C(C(CC)n2cncn2)=O)CCC(CC)CC1C(=O)NCc1ccc(F)cn1 N1(C(C(C)OC(C)=O)=O)CCSCC1CC(=O)NCCC(C)C N1(C(C(c2cc(F)ccc2Br)C)=O)CCn2c(C3CC3)nnc2C1 C1(CNC(c2nc(C)sc2C)=O)CN(C(=O)COCC2CCOC2)C(C)(C)C1 CCN=c1[nH]c(C(N2CCCC(CNC3CCC(C)(NC)CC3)C2)=O)cs1 C1(C(C)(C)C)CCC(CNC(=O)Nc2cccc(-c3cnn[nH]3)c2)CC1 C1(CNC(C2CC2CF)=O)CC2CCC1N(C(c1occc1C1CC1)=O)C2 N1(Cc2cn(CC(=O)N(C(C(N)=O)C3CC3)C3CC3)nn2)CC(O)CCC1=O N1(C(c2nc(C)sc2C)=O)CCC(C)(C)C1C(=O)NCCCC(=O)NC1CC1 c1(NCC2N(C(CNC(=O)C(F)=CC3CC3)=O)CC2)cc([N+](=O)[O-])c[nH]1 c1(C(N2CCCCC2c2n[nH]c(C)n2)C(=O)NCCOCC)cnc(SC)n1C C1(CCC)(NC(C2CC2C)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1 CC(C)(O)C(F)(F)C(=O)NC1CCCC1NC(c1cc(F)ccc1N)=O N1(C(c2cc(C#N)c[nH]2)=O)CCOC2(C1)CN(C(c1ccccc1COC)=O)C2 C=CCC(C)(C)C(=O)N1CC2C(N(C(=O)CN3CCC3C)Cc3ccccc3)C2C1 C12(CNC)CCC(CC1N)C2.c1(OC)ccccc1C(=O)N1CC1.C12CC1SC2 c1(SCC)ccccc1C(N1CC2C(C(=O)NC(CO)CO)C2C1)=O C(C(C)CC(F)(F)F)NC(C1(c2ccc(C)nc2)CCCC1)=O c1(C(C)NC(=O)N(CCOC)Cc2cccc(Br)c2)cccc(F)c1F c1(OC)cccc2c(C(C)NCc3cccc(OC)c3F)cccc12 Cn1nc(C(=O)NC(C)(C)COCCCNC(=O)C(C)(C)CF)cc1F N1(C(=O)OC(C)(C)C)Cc2n[nH]cc2C1C(=O)NC1CN(C(N)=O)C1 c1(C(=O)OC)cc(S(=O)(=O)Nc2ccc(Cl)c(Cl)c2)n[nH]1 N1(C(c2c(-n3cccn3)cccc2F)=O)CCN(C(=O)C2CC2)CC(CO)C1 N1(C(c2c(OC)cccc2)C)CC(CNC(=O)CCCn2cccn2)OC(C)C1 CC1CN(C(=O)C=CC2CCC2)CC(C)N(C(=O)Cn2cc(C(F)(F)F)cn2)C1 C1(CNC(C(F)=C(C)C)=O)CN(C(C2CCOCC2)=O)CC2(CCC2)O1 c1(C(=O)NCC(CN(C(=O)CC2CC2)C)(C)C)c(Br)ccc(Cl)c1F c1(C(N(C(C=C)C)C)=O)cc(CNC(=O)C(C)C2CCCO2)cs1 C=CC(CCC)CC(=O)N(CCCCN(C=O)C1CC1)C.c1(N)c(C)ncnc1C c1(C(N(C2CC(NC(=O)Cc3cn[nH]c3)C2)C)=O)cc(Cl)cn1C Cc1ncc(C(=O)NCC(C)CNC(C2CCC(C)C2)=O)n1C N1(C(c2ccn(CC)n2)=O)CCN(C(=O)C(c2ccc(N)cn2)C)CC1CSC c1(CC(C(=O)O)NC(=O)Nc2ccncc2Br)cnc2ncnn2c1 N1(Cc2cccc(CC)c2)CCOC(C)C1c1nc(C2CCOC2)no1 c1(C(=O)NC(CC(C)NC(=O)CC2OCCC2C)C)cc2cc(F)ccc2s1 CCC(C(=O)NCC1(C(=O)NCCc2cc(C)no2)CCCO1)SC N1(C(=O)CC(F)(F)Cl)CCCC(O)(Cn2cc(CCn3cncn3)nn2)CC1 C1(CC)CCN(C(c2sc(F)cc2C)=O)C1C(=O)NCC(C)(C)OC(C)C N1(C(CCOCC)=O)CCC2CCN(C(c3ccnc(CC)c3)=O)CC2C1 Cc1nc(CC(=O)NCC2CCCCC2NC(=O)CC(F)F)c(C)s1 c1(CC)ccc(C(N2CC3CC3C2CNC(C2CC(C)=NO2)=O)=O)nc1 c1(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)ccc(C(C)(C)C)cc1 CON(CCC(=O)NCC1CCC(=O)NC1)C(=O)C(C)N1CCC2CC12 C1(NC(COCc2cc(C)no2)=O)CCCC(NC(=O)CCC2CCOC2)C1 Cc1ccc(Br)c(C(N2CCCC(N(C)C(c3c[nH]nc3C3CC3)=O)C2)=O)c1 c1(CC(=O)NC(C(C)(C)C)CNC(c2ccsc2Cl)=O)ccc2c(c1)CCCO2 Cc1cc(C)c2cc(C(N3CCC(C4CCNC4)C3)=O)[nH]c2c1 c1(C(=O)NCC2C(CNC(C(C)(C)c3cnsc3)=O)C2)ccc(C(N)=O)cc1 C12(C(N3C(C)C(NC(C45CC(F)(C4)C5)=O)CC3)=O)CC1COC2(C)C CCCC(C)CC(=O)N1CCC(NC(C2(COC)CC=CC2)=O)C(O)C1 c1(OC)ccc2c(c1)CCCC(NS(=O)(=O)c1cc(Br)ccc1Br)C2 c1(C(N2C(CNC(CC3(OC)CC3)=O)CC(F)(F)C2)=O)cc(C)c2n[nH]cc2c1 c1(C(=O)NCC(CC(=O)NCCc2cncnc2)O)nccc2cc[nH]c12 N1(C(COC(C)=O)=O)CCC(CC(C)NC(=O)CC2COCC(C)O2)CC1 C(=O)(C(F)C(C)CC(C)(C)C)N1CCCN(C(CC(C)(C)OC)=O)C(C)C1 c1(C(CC(=O)NC2(CO)CN(C(CCC#C)=O)C2)C)ccc(N)cc1 Cc1nc(N2CCC(N(C(=O)C(C3CCCC3)OC(C)C)C)CC2)ncc1Cl CCC(CNC(N1CCC(Cn2cc(C)nn2)C1)=O)CCO.C(C)(=O)N c1(C(=O)NCC=CCNC(=O)CC2(O)CCC2)c(Br)nc2n1CCC2 N1(C(c2cc(C)sn2)=O)CCCC(NC(c2ccccc2Cl)=O)C1 CCC(C)C(C)CNC(=O)C(N1CCC(CNC(=O)Cc2ccccc2)CC1)=O CCCCCC(C)CC(=O)NC1COCC1NC(c1csc([N+](=O)[O-])c1)=O C1(C)(CNC(CN(C(C)C)C)=O)CC(F)(F)CN1C(=O)CCc1ccc(F)nc1 CN1CC(O)CC1C(=O)NC1(CNC(c2ccc(CO)cc2)=O)CCOC1 CCC(c1ccc(C)cc1)=CC(=O)NC1CCN(C(=O)C(C)(O)C(C)C)CC1C C1(NC(C2CC2C2CC2)=O)CN(C(c2cc(-c3ccc(F)cc3)no2)=O)CC1O C(=O)(CCC(F)(F)Cn1cc(CCC2CCCO2)nn1)NCC1CCC(=O)NC1 C(=O)(C1=C(C)CCOC1)NC(CC=CC)C(=O)NC1CC1CCOC Cc1cccc(N(C(=O)C(C)C(C)C)C(C2CCCN2C(=O)CC(C)(C)O)C)c1 CCCCCC(CC)C(=O)NCC1CCN(c2ccnc3nc(C)nn23)CC1 C1(NC(CCc2nc(C)c(C)o2)=O)CCC2(CC1)CN(C(C1CC1C(N)=O)=O)C2 N1(C(N2C3CCC(C3)C2c2ccccc2)=O)CCCc2c(Br)cccc21 C1(NC(c2n[nH]cc2Cl)=O)CCC(C(=O)Nc2sccc2-c2ccccc2)C1 N1(C(c2c(C#C)c[nH]n2)=O)CC(CNC(c2cnc(N(C)C)cn2)=O)CCC1C c1(C(=O)NCC(CC=C)NC(c2cnc(C3CC3)o2)=O)nccc(Cl)c1Cl CCCCCC(CCCCC)CC(=O)NC(CNC(c1occc1Cl)=O)CC N(C1CCOc2cc(OC)ccc21)C(c1cnn(CCCC)c1C)=O CN1CCCC12CN(C(C13C(NC(C4CC5CC4CC5=O)=O)C4CC1C3C4)=O)C2 CCC(CN(C)C)C(=O)N(C1CCN(C(=O)COc2ccc(F)nc2)C1)CC Cc1ccc(NC(=O)CCCCCCl)c(NC(C2CCCN(C3CCCC3)C2)=O)c1 N1(C(c2ncc(C)nc2)=O)CCC(NC(=O)CCC2(C)CC2(F)F)CC1C CC1CCCc2cc(C(=O)NCCC3CCCN(C(C4CC4(F)F)=O)C3)nn21 C12(CO)CN(N3CCCC(N4CCC(OCC(F)(F)F)CC4)C3)CC1CCO2 O=C(CCC(F)(F)Cn1cccn1)Nc1ccc(F)c(Cl)c1 N1(C(CCNC(c2ccc(C)nc2)=O)=O)CCCC2CN(C)CC12 C(=O)(CCCS(C)(=O)=O)NCCN(C)C(C1(C#N)CCC(=O)CC1)=O c1(-c2c(OC)cccc2)cc(=NC(=O)C(N)C(C)C2CCCC2)[nH][nH]1 n1(CC#C)cc(NC(C2CSCN2C(C2CCC2C)=O)=O)cn1 C#Cc1cccc(C(N2CCCCC23CC3)C(=O)NCc2ccc(F)cc2)c1 N1(C(CC2C(CC)C2(F)F)=O)CC(N(C(c2[nH]c(C)cc2C)=O)CC)C2(CC2)C1 CCC(F)(F)CCNC(=O)CCN(C(=O)CCc1ccoc1)CCO c1(-c2scc(NC(c3c(OC)cc(Cl)nc3)=O)n2)c[nH]c2ccc(OC)cc12 N1(C(CCc2onc(C)n2)=O)CCC(F)(CNC(C2CCCCC2C)=O)CC1 Cc1cc(C(C)C(=O)NC2CC(F)(CNC(C3C4CCCC34)=O)C2)cc(C)c1 c1(C(=O)NCC2(C(N)=O)CN(C(C=CCOC)=O)C2)ccc(C2(O)COC2)cc1 c1(C(N(CCCCC=C)C)=O)cccc(-c2cccs2)c1 C1(C(=O)NCC2(CSC)CCC2)CCC(O)CN1C(c1cccc[n+]1[O-])=O Cc1nnc(O)c(C(N2CCC(NC(c3ccc(Cl)cc3O)=O)C2)=O)c1C C(C(O)CC(=O)N1CC(C)(C)C1c1cn(CCC(=O)OC(C)(C)C)nn1)N(C)C Cc1ccc(C2=NOC(CN3CCN(c4nc5ccccc5[nH]4)CC3)C2)cc1C c1(CNC(C(=O)NCC2(c3ccccc3)C(C)(C)C2)=O)cc(F)ccn1 N1(C(C)=O)CCOC(C(N2CCC(CCNC(c3ccc(Cl)cn3)=O)CC2)=O)C1 c1(OC)ccc(-c2nc(CS(=O)(=O)NCC3CC3N(C)C)cs2)cc1 c1(C(=O)NC(CC)CNC(=O)Cc2csc(Cl)n2)cccc2occc12 c1(NC(N2CCCC(CN(c3ccc(Cl)cc3)C)C2)=O)cnn2cccnc12 C(C)(CN=c1[nH]cnc2c1COC2)N(C(c1n(CC)nc(C2CC2)c1)=O)C1CC1 Cc1cc(C(=O)NCC(C)CN(C)C(c2cnc(C)cc2C)=O)cc(F)c1 N1(CCN(C(C(F)OC)=O)C)CCN(C(=O)CC2CC(C)=NO2)CC1 C1(C(=O)NC2(C(=O)NCC3CC3Cl)CC2)CCCCCCC1 N1(C(CCC2CC(NC(C(C(C)C)SCC)=O)C2)=O)CCN(C)C2(CCC2)C1 C(CC1=CCN(C(c2cc(C(C)C)ccc2C)=O)CC1)NC(C=CC(C)=O)=O N1(C(C2CC3CCC2C3)C(=O)NCCC)CCC2(CC1)OCC(O)C2O CN1CCCCC1CCC(N1CC2C(C1)N2C(c1ccc(F)cn1)=O)=O N1(CCCC(=O)NC2C(CNC(C3(C)ON=C(C)C3)=O)CC2)C(=O)CN(C)C1=O n1(CC(=O)Nc2c(Cl)ccc(CC(N3CCCC3)=O)c2)nc2c(n1)CCCC2 C#Cc1ccc(F)c(C(=O)NCc2nocc2C(=O)NC2CCOC2)c1 C1(C)(N(C)C)CCCN(C(=O)CC=CCNC(=O)CC(C)(C)N(C)C)C1 C(=O)(C(C)(C)CC(=O)NC1CN(C(c2nc(C)oc2C)=O)CC1OC)OC CC1(C)CCC(NC(C23CCC(CC2)CC3)=O)C(CNC(C2(F)CC2)=O)C1 C1(NC(=O)CCn2cnnn2)CCC2(CC1)CC2N=c1nc(CC2CC2)[nH]s1 c1(C(=O)NC(CC)CN(C)C(C2CCCN2CC(C)C)=O)ccc(C)c(C)c1N N1(C(Cc2c(C)occ2)=O)CCC(C2(NC(C3CCNC(=O)C3)=O)CC2)CC1 CC1CCCCCC1NCC1CNCC1C(C)(C)C C1(C(=O)NC2CC3CN(C(c4c(N)cccc4F)=O)CC23)CC1C1CCCCC1 c1(C(=O)NC(Cc2cnc[nH]2)C(=O)NCC2CCCS2)ccc[n+]([O-])c1 c1(NC2CCN(C(CN(CC)CC)=O)C2)nc2cccc(C)c2o1 c1(COC(C(c2ccc(Cl)cc2)OC)=O)cc2n(n1)CC(C)(C)CO2 C1(C(=O)NCC(C(C)(C)C)NC(C(C)Cc2ccco2)=O)C2CCCCCCC12 c1(C(C)C)cnn(C)c1C(=O)NCCC1CC(NC(=O)Cc2ccccc2Cl)C1 N1(C(c2c(C)cccc2)=O)CC2C3CCC(C2C1)N(C(C1CNC(=O)N1)=O)C3 c1(CC(N2CCN(C(C3(Br)CCC3)=O)CC2)=O)ccc(F)cc1 N1(C(CSC(C)(C)C)=O)CC2OCCN(C(=O)CCS(C)=O)C2C1 c1(OC)cc(OC(c2cc(Br)cn(C)c2=O)=O)c2cc(C#N)ccc2c1 n1(CC(N2CC(CN(C)C(C3CC(C)(O)C3)=O)C2)=O)c(=O)oc2ccccc12 N1(C(CNS(CC)(=O)=O)=O)CCC2(CCC2)C(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 C1(N=[N+]=[N-])(C(=O)NCC(CCOC)(C)C)CCN(C(C2CC3CCC2O3)=O)C1 Cc1nn(-c2cnn(C)c2)nc1C(=O)NCCN(C(=O)C(C)(F)F)C c1(C(N2C(CCNC(=O)C(F)C3CCC3)CCC2)=O)cccc(C2CC2)c1Cl C1(C(N2CC(O)(CN(C(CCc3c(C)ncs3)=O)C)C2)=O)OCC2CCCC1C2 c1(C(=O)NCC2(C)CCN(C(=O)CC3CC4(CC4)C3)C2)coc2c1CSC2 Cc1cc(C(=O)N(C2CCN(C(c3c(N)cccc3Cl)=O)C2)C)cc(C)n1 O=C(C1=CCSC1)NC1(CNC(c2ccc(-c3nnc(S)o3)cc2)=O)CCC1 c1(CNC(=O)NC2C(CCNC(=O)OC)CCC2)cc(OC)cc(SC)c1 C1(NC(c2cc(CCC)[nH]n2)=O)CN(C(=O)Cc2ncc(Cl)s2)C2(CCCC2)C1 CCC(C)C(O)C(=O)NC1CCN(C(=O)COC2CCN(C)CC2)C(C2CC2)C1 C1(C(N2CC(F)(CF)C2)=O)(NC(C)=O)CCc2cc(Br)ccc2C1 C1(CCC)CN(C(c2cccc(OCC)n2)=O)CCN1C(C1CCCC1C)=O N1(C(CN(C(C(C(CC)(C)C)O)=O)CC2CC2)=O)CC(C2=NOC(C)C2)C1 N1(C(c2cccc(CC(C)C)c2)=O)CCC(C)C(CNC(=O)CCCC(F)F)C1 c1(CCC(C)NC(N(CCCC)CC)=O)cccc(C)c1 C1(C(N2CCCC(NC(c3cc(NC)nc(Cl)c3)=O)C2)=O)C2CCC1(C)C2(C)C c1(N2CCCC(CNC(c3cnc4ncccn34)=O)C2)nc2c(F)cccc2o1 C12(C(=O)NC3C(CNC(c4ccc(OC)o4)=O)C3)CC3CC1C2C3O c1(C(C(=O)NC(C(C)NC(C2(C(N)=O)CCC2)=O)C)C)ccc(Cl)cc1 CC1CCN(C(C2(C(F)(F)F)CCC2)=O)CC1CNC(c1nc(O)[nH]c(=O)n1)=O CN1CC(=O)N(CC(=O)NC2(CO)CC(F)C2)C1=O C(c1ccnc2ccccc12)=CC(=O)N(CCNC(C1CC(C)C1(C)C)=O)C C12(F)CCCN(CC1)C(=O)CC1CC(C1)C(=O)NC2.c1(CC)ccc(N(C)C)s1 C(C(C)(CO)NC(=O)C(C)n1ccnn1)NC(C(C)NC(N)=O)=O c1(N2C(C)CC(NC(=O)CCc3ccccc3)C2)ccnc(S(C)(=O)=O)n1 c1(C(=O)NCCC(C)NC(=O)CC2CCOC2)cc(C(F)F)ccc1Br c1(CC(=O)NCC(C)(CO)NC(C23CCC(C2)C3)=O)ccccc1Br c1(C(=O)NCC(CC=C)NC(C2CC(OC)C(OC)C2)=O)c(F)ccc(Cl)c1F c1(C(N2CCC(C(C)(C)NC(C(C)=CC)=O)C2)=O)oc2ccccc2c1CO CC(C)CC(C(=O)N(C)CC1CC(CC2CC2)C1)OC(=O)C(C)(C)C C1(C(=O)NCC(C)(C)CC2CN(C(C3CCCCNC3=O)=O)C2)CC2CCC1CC2 CC1CN(C(C2CC(F)(CF)C2)=O)C(C)CN1C(=O)CCc1ccon1 c1(C(N(C(C)(C(=O)NCc2cc(C(=O)OC)co2)C2CC2)C)=O)ccncc1 C1(C(C)NC(c2cccnc2)=O)CCCN(C(=O)CCn2cc(Br)cn2)C1 c1(CN(C(CN(C(c2cc(CC)no2)=O)C2CC2)=O)C)ccncc1C C1(CNC(C2C(F)(C(=O)OC)C2)=O)CCC(CN(C(=O)CCF)C)CC1 N1(CC(=O)N(CC(C)NC(C2CCSC2)=O)C)C(=O)CCC1=O c1(C(N2CCN(C(=O)C=C(Cl)Cl)C(CCO)C2)=O)coc2c(F)cccc12 N1(C(c2cc(CC)n(C)n2)=O)CCC2(CC1)CC(NC(=O)CCC(F)F)CO2 c1(C(=O)NC2CC(NC(C(CC)(C)F)=O)C2)ccc(-n2cnnn2)cc1Cl N1(C(c2ccc(Br)cc2)=O)CC2CN(C(c3occc3Br)=O)CC12 c1(C(=O)NC(C(=O)NCC(O)CNC=O)Cc2ccsc2)cc(Cl)cnc1O CC1C(NC(c2cc(C(N)=O)[nH]n2)=O)CCCN1C(=O)CC=CC(C)(C)C C#CC1(CNC(=O)CC(C)CNC(c2ccns2)=O)CCOCC1 c1(C(=O)NC(CC)CNC(=O)COCC2CCC2)ccc(-c2nnc(S)o2)cc1 N1(C(C(C)CC(C)N)=O)CCCc2cc(N3CCNC3=O)ccc21 C=C1CC(C(=O)OC(C)(C)C)(CNC(=O)C(C)NCC2(F)CCC2)C1 C1(F)(CNC(CN(C2CCSC2)C)=O)CC(CNC(c2ncoc2C(F)F)=O)C1 CC1(C)C(C)(C)C1(F)C(N1CCC(C(=O)NCc2cn(C3(C)CC3)nn2)CC1)=O Fc1ccc(OCCNCc2cncs2)cc1C1CCCCC1 c1(CC)occc1C(=O)NCC1CC1NC(=O)CCN(C)CCO c1(CC)nc(C(=O)NCC(CC2CCCO2)OC)c2n1CCCC2 c1(C(=O)OC)cnc(O)c([N+](=O)[O-])c1.c12ncc(nc1C)NCC(O)CNC2=O C1(C)(CCC)CCCN(C(=O)C(CC(F)F)N(C)C(c2sccc2CO)=O)C1 N1(C(C2N(CC)CCOC2)=O)CCN(C(C23COCC(C2)C3)=O)CC(O)C1 N1(C(CN(C(C=C(COC)C)=O)C2CC2)=O)CCOCC12CC2 c1(OC)ncccc1C(=O)NC1(CF)CN(C(=O)Cc2cc(C)cs2)C1 c1(OCC)cc2cc(C(=O)NCCc3ccnc(OCC)c3)[nH]c2cc1OC c1(C(=O)NC(CC=C)CNC(c2ccsc2Br)=O)cccc(CC)n1 C1(CC(N2CCCC2)=O)CC2CCC1CC2.N12CCCC(C1)CNC(=O)C2 c1(C(=O)NCC2(NC(C3C(=C)C3)=O)CCOCC2)cc(S(N)(=O)=O)ccc1O c1(NC(C2CCC2)=O)nc(C)sc1C.Cc1ccsc1CN1C(=O)C1C1(C)CC1 C1(C(N2CCC(C(N3CC(C(C)C)(CO)C3)=O)C2)=O)CCCC(C)(C)C1 CC(O)(CNC(c1occc1CNC(C1COCC1C(N)=O)=O)=O)CO C1(CNC(c2ccoc2)=O)CN(C(=O)CCCn2ccnc2)CC12CC2 c1(C(=O)NC2C(C(=O)NC3(C(=O)NCC)CC3)CCC2)cncc(CC)c1 C1(O)(CCNC(COCC(=C)C)=O)CN(C(=O)NCCS(=O)(=O)CCC)C1 C1(NC(N(C)Cc2ccc(C)nc2)=O)CC[Si](C)(C)CC1 N1(C(c2ccccn2)=O)CCC(CC(CN)CO)CC1 c1(C(=O)NC(C)CNC(=O)C(O)C(C)(C)C)ccc2c(c1)C=CS2(=O)=O CN1CCN(C(=O)CCc2ccncn2)CC1CNC(=O)CC(F)(F)Cl c1(C(=O)OC)cc(Cl)c(NC2(CCNC(C3CC(=O)N(C)C3)=O)CCC2)nc1C N1(C(C=CC=CCCCCC)=O)CCC(C)(CCNC(c2ccnc(C)c2)=O)C1 C1(C(N(CC(CN(C(c2c(C)noc2)=O)C)O)C)=O)Nc2ccccc2C1(C)C Cc1cc(N)c(C(N2CCC(C(C)NC(c3cc(C4CC4)no3)=O)C2)=O)cc1F c1(C(=O)OCC)cnc2sncc2c1NC1COc2cc(Cl)ccc2O1 c1(C(N2CC3(N(C(C(CCC)C)=O)CC3)C2)=O)cn2cccc(Br)c2n1 N1(C(C(C)=C(C)C)=O)CCCCC1CCN(C)C(C1C(Cl)(Cl)C12CC2)=O N1(C(c2cc(OC)no2)=O)CC2CCCC1C2CO N1(C(CNC(C)=O)=O)CCCC(C)(C(=O)NCC(c2ccccn2)C)C1 N1(C(C(CC)CC)=O)CCN(C(=O)CC(O)C2CCCC2)C(CC(F)(F)F)C1 C(c1ccc(Br)nc1)=CC(=O)N(C1CCN(C(C(C=C)(C)C)=O)C1)CC CCC(C(=O)NCc1cn(C2CN(C(c3cc(Cl)n[nH]3)=O)C2)nn1)OC C=CCCC(C)N=c1[nH]c(=NCC2CCCSCC2)[nH]c2cc[nH]c12 C1(C(C)C)CCc2sc(C(=O)NCC3CCN3C(=O)CCCC(N)=O)cc2C1 c1(CC)nc(C)[nH]c1C(=O)NC(C)CN(C)C(c1n[nH]c(C)c1Cl)=O C1(CC(=O)N(C2CCOC2)C)CC(F)CN1C(=O)CC1CCOC1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCN(C(c2cc(OC)n[nH]2)=O)C1(C)C n1(CC(N2CCCC(NC(CNC=O)=O)C2)=O)nc2n(c(=O)c1=O)CCOC2 Cc1cc(C(=O)NC(CNC(=O)CC(O)C2CCC2)C2CC2)n(CC(F)F)n1 C1(C(=O)NCC#C)CN(C(C2CCC(=O)C2)=O)CC1CCC c1(CC)conc1C(=O)NCCC(CNC(=O)C(C)Cc1ccncc1)OC c1(CNC(CC2C(CN)C2)=O)ccn2cncc2c1 c1(C(N2CC(O)(C(C)NC(=O)C3=CCCCC3)C2)=O)cnc2n1CCCC2 c1(C(=O)NCCOCCNC(CCN(C)CC)=O)ccnc2c(F)cccc12 c1(OC)nc(C)ccc1C(=O)NCC1(C)CCCN(C(=O)C2=CCOC2)C1 c1(C(=O)NC(C2CN(C(C3CC3C)=O)C2)C)cncc(-n2cccn2)n1 c1(C(N2C(C)CCC(NC(c3cnco3)=O)C2)=O)ccc2nccn2n1 N1(C(C2C(C(=O)OC)C2)=O)CC2CC1CC2CNC(=O)CSc1cnn(C)c1 N1(C(c2cc(C)nc(C)c2)=O)CC2(CCCC2)C1C(N1CC(CN(C)C)C1)=O C1(C(N(CCCC(=O)NC(C#C)(C)C2CCC2)C)=O)CCC(C)(C)CC1 N1(C(C2C(C)(C)C(O)CC2)=O)CC2(COC(CNC(=O)OC(C)(C)C)C2)C1 C1(NC(CCc2n(C)cnn2)=O)CC(NC(c2ocnc2C(F)F)=O)C(O)C1 c1(C(N2CCC(OCCNC(C3C(OCC)C3)=O)C2)=O)cc(N)nc(Cl)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(C)=O)C(C)C1 N12CC(C)(C)C1C2=O.C=C=CCC(=O)N1CSCC1C(=O)NOCC CCCCCCCCC(=O)NC12CCC(C1)N(C(c1ccc(C(N)=O)s1)=O)C2 c1(C(N2CCC(C)C(CNC(c3nc(Cl)cs3)=O)C2)=O)ccnc2cc[nH]c12 C12(C(N(CCOC)CCNC(=O)CCC3CC34CC4)=O)CCC(CC1)C2 C12(NC(C(C)NC(=O)NC)=O)CC(C)(C1)OC21CN(C(C2(SC3CC3F)CC2)=O)C1 CCCCCCCC(C(=O)NCCCOC)N(C)CC1CCN(C)C1 CN1CCN(C)C(C(=O)NCCCOCCNC(=O)C2=COCC2)C1 C1(C)(C(=O)NC(c2ccc(Cl)cc2)C(C)C)CCN(Cc2cnco2)C1 CC(C)C(CNC(=O)C(C1CCOCC1)C)C(=O)NCCN=S(C)(C)=O c1(C(=O)NCc2nncn2-c2ccccc2)cnc(C2CCC2)nc1O N1(C(C=CC)=O)CCC(NC(=O)C=C2CCN(C)CC2)C(O)C1 Cn1ccc2c(C(N3CC(NC(C4CC(F)(CO)C4)=O)CC(O)C3)=O)ncnc12 c1(CN(C(=O)NCc2cnc(COC)s2)C)ccc(OC)cc1Cl N1(C(C(C)N(C)CCNC(=O)Cc2ccnn2C)=O)CC(C)OC(C)C1 C1(CC(=O)OCC(C)(C)CC2CCCCC2)(CNC(=O)OC)CCOCC1 c1(C2(Cc3nn(-c4c(C)cccc4)c(C(C)CSC)n3)CC2)c(F)cccc1F N1(C(CC(C)CF)=O)CC2CN(C(c3nocc3Br)=O)CC2C1 N1(C(c2nc(C#C)sc2)=O)CCCC(NC(C2CC=CCC2)=O)C1C CCCC(C(=O)NCCN(C)C(=O)C1CC1)NC(C1CC1C(C)C)=O c1(C(=O)NCCN(C(=O)C=CC2CC2)C)cncc(C(=O)OC(C)(C)C)c1 c1(C(=O)NC2CCN(C(C3(C)CC(C)C3)=O)CC2O)noc2c1CCCC2 c1(OC)ccc(-c2cn3cnc(C(N4CCC(Br)C4)=O)c3s2)c(F)c1F CC(=O)CCC(=O)NCC(C)CNC(c1cncc(Br)c1)=O C12(NC(=O)C(O)C3CCC3)CCCC1(F)CN(C(=O)C=CC1CCCCCC1)C2 c1(CC(=O)NCC(CC=C)NC(C23CCCC2C3(F)F)=O)cc(Cl)cc(Cl)c1 CC(C)C(C(=O)NCC1C2CN(C(=O)CN(C)C3CC3)CC12)NC(=O)C(F)(F)F c1(NC(C2CCC(NC(=O)Nc3ccc(OCC)cc3)C2)=O)c(F)cncc1Br N1(C(CCCn2c(C)ncc2)=O)CCC(C(C)(C)NC(=O)CC2CC2(C)C)CC1 c1(OC)cnc(CNC(=O)C(O)CNC(=O)CN2CCCCC2=O)cn1 CCCC(CC)CC(=O)N(C(CNC(=O)C(=O)N(CC)CC)CC)C c1(C(=O)NC(C)CN(C(=O)C(C2CC2)OC2CCCC2)C)nnn2c1COCC2 Cc1ccc(Br)cc1NC(C1(F)CCCN(C(c2cccc(F)c2F)=O)C1)=O C1(C(=O)NCC=CCCC)CCCCN1C(=O)CCNC(=O)CO C1(CNC(C(CCC)OC)=O)CCN(C(=O)CCc2ccc[nH]2)C12CCC2 Cc1cc(C(=O)NC(C2CCCC2)CNC(=O)C(C)NC(=O)C(C)(C)C)no1 N1(C(CC(C)CN(C)C)=O)C2CCC1C1CC1(NC(=O)Cc1nncn1C)C2 CC1CCCN(C(=O)CCS(N)(=O)=O)C1CCNC(C1CC(OC(F)F)C1)=O C1(CC)CN(C(=O)CC(C)C)CCC1NC(=O)CCCNC(c1ccccn1)=O CCCC(CNC(C1(NC(=O)CC2CCC(C)CC2)CC(F)(F)C1)=O)CCO c1(CC)ccc(C)nc1N1CCCCC1C(=O)Nc1cn(CCCOC)nn1 Cc1nn(CC(C)C)c(C)c1CC(=O)NCC(O)CNC(=O)CCCC(F)F C(C)(CC(=O)NCC1CCCN1C(=O)C=Cc1ccsc1)(C(F)F)N(C)C c1(-c2n(C(CCNCC(F)(F)F)c3ccco3)ccn2)ncc(-c2ccccc2)o1 CCC(C)C(C)C(=O)NC1C=CCCC1C(=O)N(CCCC(=O)NC)C Cc1ccc(C(=O)NCCN(C)C(c2cc(C3CC3)[nH]n2)=O)c(=O)n1C N1(C(=O)CC(F)(F)F)CCC(C2CCN(C(=O)CCC(=O)c3ccc[nH]3)C2)C1 N1(C(CNC(C(CC)C)=O)=O)CC(NC(C2(C)COCCO2)=O)C(C)C1 c1(C(=O)NCCCOCCNC(C2CCCO2)=O)cnn(C2CCCC2)c1 N1(C(C(=C(C)C2CC2)F)=O)CCCC1CNC(=O)CCCNC(=O)NCCCO C1(C(=O)NC(C#C)C)COC2(CCN(C(c3ccc(C)cc3Cl)=O)CC2)C1 C1(CN(C(COCC(=O)OC)=O)C)CCCN(C(=O)CCCNS(C)(=O)=O)C1 c1(CNC2COC(F)(F)OC2)c[nH]c2ccncc12 C=CCCCC(C(=O)NCCOC(C)C)NC(c1cc(O)ncn1)=O c1(C(C)C)nccc(C(N2CCC(N(C(=O)CC3CCC(=O)N3)C)CC2)=O)n1 O=C1CN(C(=O)CC2CCCCC2NC(C23CCC(OC)C2C3)=O)CC(=O)N1 CC1CCCC=C1C(=O)NC(C1CCCC1)CNC(c1cnc2ncccn12)=O CC(C(=O)N1CCC(C2(C(F)(F)F)N=N2)CC1)C(F)F C1(OC)CC(NC(C2(C#N)CCC2)=O)CN(C(=O)C(c2cccc(C)c2)(C)C)C1 C1(C(N(CCOCCNC(C=C(C)C)=O)C)=O)CCN(C)C1 N1(C(CNC(=O)NC)=O)CCCC12CN(C(c1cnc(OC)cc1OC)=O)C2 c1(C(=O)NCC2C(CNC(C(CC)N(C)C)=O)C2)csc2ncnc(O)c12 N1(C(C(CC)N(C)C)=O)CCC2(CCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 C#Cc1cc(C(=O)NC2(C)CC(NC(=O)CSc3nccn3C)C2)cc(Br)c1 C1(CNC(C(CSC)(C)C)=O)COCCN(C(=O)CCN2CCCC2=O)C1 C1(C(=O)NC(CCC)(C)CC)CC(c2ccc(Cl)cc2Cl)=NO1 C(=O)(N1CCCCCO1)C1(CN(C(c2cncc(C=C)c2)=O)CC)CCC1 CCC(CC)CCC(C(=O)NC1CCC1)N1CC(CO)C(C2CC2)C1 c1(C2(C(N(C3(c4nnnn4C4CCCC4)CC3)C)=O)CCC2)ccccc1Cl N1(C(CCOC)=O)CCCC1C1CCCCN1C(=O)Cc1cc(C)ns1 N1(C(C2C=C(C)CS2)=O)CCC(NC(c2cc(C)nnc2O)=O)C(C)(C)C1 CN1C(=O)CSC1=CC(=O)NC(C)(C)CCNC(=O)CC1CC(O)C1(C)C C12(CNC(C3(COC)CC3)=O)CC(NC(C3CCC3C)=O)(CCO1)C2 C1(C(=O)NCC2CC(NC(CS(CC)=O)=O)C2)CCN(C2CC2)S1(=O)=O CC1(C)CC(NC(=O)CC2CCC(F)(F)CO2)CN(C(=O)C(C)(C)C#N)C1 c1(C(=O)NCC(CN(C(Cn2nc(C)c(Cl)c2C)=O)C)O)c(F)ccc(N)c1F c1(C(=O)NCCN(C(C2(C#C)CC2)=O)C)cc(S(N)(=O)=O)n(C)c1 c1(OCC)ccccc1C(=O)NC1CCC(NC(=O)CC2CC(OC)C2)C1 Cc1nc(CC(=O)NC(C)(CNC(=O)C(C)CN(C)C)CO)c(Cl)s1 N1(C(Cc2cccc(C)c2)=O)CCCC(CC(=O)CCN2CCCCCC2)CC1 C1(NC(C(CCC)C)=O)CCN(C(c2ccc(C)nc2N)=O)CC(C)(C)C1 C1(NC(C(CCNC(C2(CC)CCCC2O)=O)OC)=O)CN(C)C(C)(C)C1 C#Cc1cnc(C(=O)NCC(C)CC(=O)N2CC(OC)CC2C(N)=O)c(C)c1 C(Cc1cn[nH]c1)(C(=O)NC(c1csc(C)n1)C)NC(C1C(C(=O)OC)C=C1)=O C(CCC(CO)NC(=O)CC1CC(=O)NC1=O)CNC(C)=O C1(C(=O)NC2(C)CC(NC(C3(COC)CC3)=O)C2)CCC(=O)N(C(C)C)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCCC(C)N(C(CCNC(=O)NC)=O)C C1(CSC)CCC12CCOCC2.C1CCOCCOCCNC(=O)N1 N1(C(COCc2c(C)nns2)=O)CC(NC(=O)C(C)(C)CF)C2CC12 Cc1ccccc1NCC(=O)N(CC(C)N(C)C(c1cnncc1O)=O)C c1(OCCC)ccnc(N2CCC(NC(=O)CSc3ccccc3)C2)n1 CN1CCCCC(C(N2CC(O)(CCNC(=O)COC(F)F)C2)=O)C1=O C1(C(N2CC(CNC(C(C3CCCC3)OCC)=O)C(C)C2)=O)CC(C)OC(C)C1 c1(OC)c(NC(C)CCNC(c2ccc(Cl)nc2C)=O)ncnc1C CC1(C(=O)NC2CCC(NC(c3csc(C(F)(F)F)n3)=O)C2)CCNC1=O c1(-c2scc(NC(c3c(C)cc(I)cc3)=O)n2)cccc(F)c1C#N c1(C2CC(C(N3CC(NC(C4(F)CC=CC4)=O)C3)=O)C2)ccc(F)cc1 C(=O)(C(C)(C)C(=O)OC1(C(=O)NC(C)(C)C)CC1)NC(CC(C)C)CNC(C)=O C1(O)(C(C(N2C(C(C)(C)C)CCC2)=O)NC(=O)C=CC(=O)NC2CC2)CCCCC1 C1(CC)C(C(N2CCC(O)CC2)=O)CCN1C(c1ccc(CO)cc1)=O c1(C(=O)NCc2cccc(C(C)(C)C)c2F)cc(-c2nn[nH]n2)cc2c[nH]nc12 C(=O)(C1SCCc2ccccc21)N1CCC(C)(NC(CC(=O)N(C)C)=O)C1 CC1CCCC1(C(=O)NCc1cn[nH]c1)NC(=O)C=C1CCSCC1 C(=O)(CC1=CCN(C(=O)C(C)(F)F)CC1)N1CCCC(OC(C)C)C1 c1(C(=O)NC2CC(C)N(C(=O)C#CC(=O)N(C)C)CC2)cnc2n(c1=O)CCS2 c1(SC)nc(=NC2CN(C(=O)Cn3ncc(O)nc3=O)Cc3ccccc32)s[nH]1 N#CC1CN(C(=O)C=CCn2ccnc2)CCN1C(=O)Cc1ccc(F)cc1 C(C)(CCC(=O)NCCCN(CCCNC(c1cc(Cl)ns1)=O)C)SC c1(CNCc2cnc(CC)[nH]2)ccc(S(N)(=O)=O)o1.N12CCC(=CC1=O)CC2 c1(OC)cc(C(=O)NCCCNC(=O)CCc2ccccc2O)c(F)cn1 C(C(N=c1[nH]c(NC2CN(C3CC3)CC2C)nc2ncn(C)c12)C1CC1)OC C1(NC(c2cc(C)c(F)cc2)=O)CCC2CN(C(c3cc(Br)c[nH]3)=O)CC2C1 CC1=NNC(=O)C1CCC(N1CC2CC2(CNC(c2[nH]c(C)nc2C)=O)C1)=O C(CCNC(=O)C(C1CCC1)C1CCC1)(C(C)C)NC(C1(CC#C)CCCO1)=O Cc1ccc2c(c1)CC(C(N1CCC(N(C)C(c3ncncc3Cl)=O)C1)=O)S2 N1(C(=O)CCCN2CCNC2=O)CCCC(n2cc(-c3nccc(Cl)n3)nn2)C1 C1(NC(=O)Cn2cnnn2)CCN(C(c2n[nH]c3c2COCC3)=O)CC12CCC2 c1(C(N(C(CNC(C(CC#C)C)=O)C)C)=O)cc2cccnc2nc1C1CC1 N1(C(C2C(C(N)=O)C2)=O)CC(NC(C23CCCC2C3)=O)C(n2cccn2)C1 C1(CC(=O)NCCCCn2cc(COCC(N)=O)nn2)CC(O)C1(C)C c1(C(N2C3C(CNC(C(CC)SC)=O)C(C3)C2)=O)ccc(N)c(N)n1 c1(-n2cc(CC(C(=O)NCCCCN3CCCC3)O)nn2)ccc(Cl)c(F)c1 C12(C(=O)NC(C(C)F)C)CC1CCN2C(c1cnsc1)=O C(=O)(CC(O)C(C)(C)C)NCC1CCN(C(CN(C)C2CC2)=O)CC1 c1(-c2nc(C(CC)CC)nn2-c2cnn(C)c2)ccnc2ccc(OC)cc12 c1(C(=O)NCCN(C2CCCC2)C(C2C(CC)C2)=O)cccc2c1OCCCC2 N1(C(c2n(CC)c(O)nc2)=O)CCC2(CC1)CC(NC(C1CCOC1)=O)CO2 CC(=O)CCN=C(NCc1cccc(Cl)n1)NC(C1CCOCC1)C C(=O)(C(CCOC)NC(c1ncsc1C)=O)NCCOC(CC)(C)C c1(CC)cccc(CC(N2CCOCC2CN(C(=O)CC(O)CN(C)C)C)=O)c1 C12(CS(C)(=O)=O)CC(CN1C(C1CC1C1CCC(=O)O1)=O)C2 Cc1cc(=O)ccn1CC(=O)NC(C)C(C)(C)NC(C1CC(O)(C#N)C1)=O Cn1cc(C(N2CC(CNC(C3CCCC3CF)=O)C(O)C2)=O)c2cccnc12 C1(CNC(CCOCC)=O)CN(C(C2(n3cccn3)CC2)=O)CC12CCOCC2 CCC(C)CCCC(=O)N1CC2(NC(c3cnc(C(C)C)nc3)=O)CCC1C2 N1(C(=O)Cn2ccccc2=O)CC2(CCN(C(C3(C4CCCC4)CC3)=O)CC2)C1 C(CNC(c1cnns1)=O)(C(C)C)NC(CCNS(CC)(=O)=O)=O C1(NC(c2c(-c3ccc(C)s3)ocn2)=O)CN(C(=O)CC2CCCCO2)CC1C c1(CC)ccc(NC(=O)NCc2cncc(OC(C)C)c2)c(Br)c1 CN1CCC(C(=O)NCC2C3CN(C(=O)C(F)(F)c4cnccn4)CC23)C1=O C(CC(=O)NCc1cn(C(C)Cc2ccc(N(C)C)nc2)nn1)(C(F)(F)F)OC CCCC(O)CC(=O)N1CCCC(NC(=O)CCCN(C)C)C1C C1(CC)CN(C(c2cc(C)cs2)=O)CCN1C(C1CC(C(F)(F)F)C1)=O c1(C(N(CC(CNC(c2cn(CCC)nc2)=O)O)C)=O)cc(F)cc(F)c1OC c1(C(=O)NC(C)CNC(C2(C)CC2(F)F)=O)csc2ccc(F)cc12 C(=O)(C(C)CN(C)C(C1CC(C)N1C(=O)CCc1ccn(C)n1)=O)OC Cc1c(C(=O)NC(C2CCCCC2)C23CNC(C2)C3)noc1-c1ccccc1 C#Cc1cn(C)nc1C(=O)OC.C12CC3CCC1N3C2 c1(CC)cnoc1C(N1CCC(NC(=O)Cc2csc(C(F)(F)F)n2)C1)=O c1(C(N(CCCN(C(=O)C(C2(O)CCCC2)F)C)C)=O)ccnnc1 Cc1ccc(C(=O)N(CCCCCCNC(=O)C(C)CN(C)C)C)c([N+](=O)[O-])c1 N1(C(CN(C(C)=O)C)=O)CC(NC(c2ncc[nH]c2=O)=O)C(C(F)F)C1 C1(NC(C=CC)=O)CCCCC12CCN(C(c1cc(C(C)C)[nH]n1)=O)C2 N1(C(C2CCN(C(c3ncn(CC)n3)=O)C2)=O)CCOC2CCOCC12 c1(C(N(CC(CNC(CSCC)=O)C)C)=O)c(Cl)csc1Cl c1(NC(C2CC23CC3)=O)cccc(OC2CN(C(CC3C(C)(C)OC3)=O)C2)c1 C1(NC(C2C3CN(C(C4C(C)(C(F)F)C4)=O)C2C3)=O)CCc2n[nH]cc2C1 c1(OCC)cccc(C(=O)NC(CNC(=O)C(=Cc2cccs2)C)CC)c1N CN1C(C(N)=O)CCC1C(=O)NC1CCN(CCNC2(NS(C)(=O)=O)CCC2)C1 C1(C(C)C)CN(C(c2cc(F)n[nH]2)=O)CCCN1C(=O)Cc1ccccc1F c1(-c2cn(CC3CN(C(CCN4C(C)CCCC4)=O)C3)nn2)cc(F)ncc1F c1(NC(c2ccc(C3CC3)o2)O)c(Cl)nsc1Cl c1(NC(C2CC(F)CN2C(=O)C(c2cccc(Cl)c2)O)=O)cccc(Cl)c1Br C1(COC)CN(C(=O)COc2ccsc2)CCN1C(C1CC2CC2C1)=O C=CCC(C)(C)CC(=O)NCC1(CNC(C2CCSC(C)C2)=O)CCCCC1 c1(CC(N2CCC3(CN(C(C)=O)C3)CC2)=O)cnn2c(C(C)O)cc(C)nc12 C#Cc1c[nH]nc1C(N1CC(OC)C(NC(C2(Cl)CC2(F)F)=O)C1)=O CC(CC(=O)N(CCCCCNC(C12CCC(C1)C2)=O)C)C(F)(F)F c1(C(=O)NCCCCNC(c2c(C3C(C)C3)noc2)=O)cnn2c1CCCC2 C1(CC#C)CCCN1C(=O)C(CSCC)NC(c1coc(C(C)C)n1)=O N#CCCCCCC(=O)N1CCC(NC(c2ccc(F)c(F)c2)=O)C1 Nc1c(C(=O)NCCOCCNC(c2ccc3c(c2)CC3)=O)ccc(Cl)c1O c1(CC(=O)NCC2C(NC(c3ccc(C)cn3)=O)C2)c[nH]c2ccccc12 C1(NC(C(C(CC)O)C)=O)CCC2(CC1)CN(C(=O)C(c1ccccn1)O)C2 c1(C(=O)NC(CNC(c2conc2C2CCCO2)=O)CO)nc(Cl)cs1 C1(OC)CN(C(=O)CC(C)NC(=O)CCC(C)C)CC1C(=O)OC(C)(C)C N1(C(c2ccccc2)=O)CCCC2(CCCN2C(c2cc3sccc3cn2)=O)C1 C(CCC(C(=O)N1CCC(O)(CO)CC1)NC(c1cc(Cl)no1)=O)OC c1(N(C(CONC(C2CC(CCC)C2)=O)=O)C(C)C)cccc(C)c1O Cc1ccc(C(=O)NC2CCCC2NC(=O)C(C)C(F)F)c(Cl)c1 c1(NCC2C3CN(C(C4(CC)COC4)=O)CC32)ncc(Br)cc1[N+](=O)[O-] N1(C(c2cscn2)=O)CCC2CCCN(C(=O)Cn3cnc([N+](=O)[O-])c3)C2C1 c1(C(N(C2CCN(C(Cc3c(C)nc(S)s3)=O)C2)C)=O)ncc(Cl)cc1F N1(C(CSCCC)=O)CCCC2(CNC(c3ccc(Cl)nc3O)=O)CC12 N1(C(CNC2CCC(=O)NC2=O)=O)CCCC2(C(c3cnn[nH]3)=O)CC2C1 c1(C(=O)NC(CCN(C(C(C(C)C)SCC)=O)C)C)ccc2c(c1)ncn2C c1(C2C(SCC)CCC2)nnc(COC)n1C(C)C c1(CC)cc(C(N2CC(C(=O)NC3C(C)C3C)CC2(C)C)=O)cc(F)c1 N1(C(C)C(=O)NC2CC(CNC(C3CC3F)=O)C2)C(=O)CCC1=O C1(NC(CCC(N)=O)=O)CC2CC(NC(=O)COc3cccc(Cl)c3Cl)C1C2 C(=O)(CC1=CCN(C(c2ccnnc2C)=O)CC1)NCc1ncc(C)o1 CC(C)(F)CCC(=O)NCC1CC(C(=O)NCCCCC2=CC=C2)=NO1 CC(CN1CCOC1=O)C(=O)NC1(CCO)CN(C(=O)Cn2cccc2)C1 C1(CC(N2C(C)(COC)CC2)=O)CCCN(C(C2(CC3CCC3)CC2)=O)C1C CC(CCC1CC1)CCNC(=O)C(C1CCCCCC1)N c1(-c2c(CNC(c3n(CC)nnn3)C3(C)CC3)cccc2)nc2ccccc2s1 c1(CC)ccc(C(N2CCCC(NC(=O)Cc3sccc3C)CC2)=O)c(C)c1 C12(C(=O)NCC3(CO)CCN(C(c4cc(C)nn4C)=O)C3)CCC(CC1)C(C)O2 N1(CCC(=O)NC(C2(O)CN(C(=O)C(C)(C)C(N)=O)C2)C)CCCc2ccccc21 c1(OC)cccc(C(=O)NC2CCN(C(=O)C(C)(C3(C)CC3)OC)CC2F)c1O c1(OC)ccc2c(c1)NC(=O)C2CC(=O)N1CCN(C(=O)C2=CCCC2)CC1 c1(C(=O)NCC(C)NC(C2(C)ON=C(C(C)C)C2)=O)cccc(P(C)(C)=O)c1 n1(CC(N2CC3C(NC(C(COC)N(C)C)=O)(C3)C2)=O)ccc(=O)n(C)c1=O CCCCC(C(=O)NCCCN(CC(C)C)C)NC(C1CC=CC1)=O c1(C(N2CCC(C(CNC(CC=CC=C)=O)(C)O)CC2)=O)cc(CC)ccc1C N1(CC)CC2CC1CN2C(c1ccc(CNC(=O)CCC(C)N(C)C)s1)=O c1(CNC(C2N(CC)CCCC2)=O)ccc(CNC(c2cccn2C)=O)cc1F c1(CC(N2CC(CCNC(CC(C(C)C)OCC)=O)C2)=O)ccc(Cl)c(F)c1 C1(C(C)C)CN(C(C2CCNC2=O)=O)CCN1C(=O)C=Cc1ccccn1 CC1(C)CC(C(=O)NCCOCC2CCC2)N(C(c2ccn(C3CC3)n2)=O)C1 CC(=O)CCCCC(=O)NC(Cn1cncn1)C(N1CCCCCC1)=O c1(CC(=O)NCCC2CC(C(=O)NCc3ccc[nH]3)C2)cnccn1 c1(C(=O)NCC2CCN(C(=O)CC3CCCCO3)CC2)ccc2ccccc2n1 c1(C(=O)NC(CNC(C2(CC)CC2(F)F)=O)CC)cccn2c(C)nnc12 C1(CC)(CC)CC(NC(c2ccc(C#N)cn2)=O)CN1C(c1ccc(SC)s1)=O C1(NC(C(N2CCCCC2)C)=O)CCCC(CNC(=O)CCOC2CCCC2)C1 N1(C(C=C(CCC)C)=O)CCC2(CCC(NC(C3(CF)CCC3)=O)CC2)C1 C1(NC(c2cc(C)sc2)=O)CC2CC(C1)CN(C(=O)CC1CCOC1=O)C2 N1(C(=O)NCCOC(C(=C)C)=O)CCCC2(CCN(Cc3csc(Br)n3)CC2)C1 C1(C(C)(O)CNC(C2CC3C=CC2C3)=O)CCN(C(=O)Cn2ccnn2)CC1 C1(Cn2cc(CCNC(N)=O)nn2)CCCCN1C(=O)CC1CCCOCC1 N1(C(c2c[nH]c(=NC)s2)=O)CCN(C(=O)Cc2occc2C)CC1C(C)C C(C(C)(C)C(=O)NCC1C2CN(C(c3cc(C)c[nH]3)=O)CC12)OC c1(-c2cn(C)nc2)ccc(NC(C2(O)CNC2)=O)nc1 C1(C(F)(F)F)(C(=O)NCCC2CC(NC(C(C)NC(C)=O)=O)C2)CCCC1 N(C(=NCC1CNC(=O)O1)n1ccnc1)CC(Cc1cccc(OC)c1)(C)O CC1CCC(NC(c2ncoc2C2CCC2)=O)CN1C(=O)C1=CCCCO1 N1(C(C(CC2CCC2)NC(C2CC2F)=O)=O)CC2CC2(CO)C1 CCC(F)(F)CCNC(=O)C(CCNC(=O)C(C)n1cnnn1)OC C1(CC(=O)NC(C(C)C)CNC(=O)CC(C)N(C)C)CCCCC1O c1(OC)cc(F)c(NC(=O)CC2(NC(c3nc(C)c(C)s3)=O)CCC2)cn1 C(=O)(C1=C(c2ccccc2)CCCC1)N1CCC(N(C(=O)C(C)N(C)C)CC)C1 C(CC1=CCN(C(C2(C)CCC(C)(C)CC2)=O)CC1)NC(CSC(C)C)=O C1(CC(N2CC(NC(C3CCC(O)CC3)=O)C2)=O)CCC2(CCC2)CO1 C1(NC(c2cnc(O)nc2O)=O)CCN(Cc2cccc(OCCF)c2)CC1F C=CC(CCC)CC(=O)N1CC(OC)C(NC(c2cc[n+]([O-])cc2)=O)C1 n1(CC)ncc(C(N2CCC(C(=O)NC3CCOC3C(C)C)CC2)=O)c1Cl C1(C(=O)NC2(CO)CCN(C(CC)=O)C2)CC12CCS(=O)(=O)CC2 C1(CC(=O)NC2C(CNC(COCCC=C)=O)CCC2)C(C)(C)C1(C)C C1(CNC(C(C)SC(F)F)=O)CCC2CN(C(c3cnncc3O)=O)CCC2C1 C1(F)(CNC(CC2(C)CC2)=O)CCN(C(C2(C)CCOC2)=O)C1 C1(F)(CN(C)C(c2cc(O)nc(Cl)c2)=O)CCN(C(=O)CNS(N)(=O)=O)CC1 c1(CNCc2c(CCC)n[nH]c2)cc(Cl)cn1C CC1CCN(C(c2cncn(C)c2=O)=O)CC1CNC(c1cc(F)n[nH]1)=O c1(NC(c2ccc(CNC(C3(CC)COC3)=O)cc2)=O)c(O)cccc1F C(C(C)(C)CC(=O)NCC1CN(C(=O)C(C)CCc2cccc(F)c2)C1)OC N1(C(CN2CC(C)C2)=O)CC2(CCN(C(c3cnc4ccsc4c3)=O)C2)C1 c1(CC)ccc(Br)cc1C(=O)NCC1CC(NC(C2(C)CC=CCC2)=O)C1 c1(C(N2CCC(COC)(CNC(=O)CC(O)CN(C)C)C2)=O)c(C)ccnc1O C1(CC)(CC)CC(C(=O)NC2(C(=O)N(CC(C)O)C)CC2C)C1 C1(C(N2C3C(NC(c4ccoc4Cl)=O)CC(C3)C2)=O)CCC2(CCOCC2)O1 N1(C(COC(C)=O)=O)CC(C)CN(C(=O)COC(c2ccccc2)C)CC1C N(C(=NCc1nocc1Br)N(C)CC1CCOC1)C(COC)C N1(C(c2c(C)nc(CC(C)C)s2)=O)CCN(C(=O)C#CC(C)C)C(C)C1 N1(CC)CCCCC1C(=O)NCC1CC(F)CN1C(c1cc(Cl)cnn1)=O c1(OC)ccc(CCC(=O)NCCCOCC(c2cccc(C)c2)=O)cc1 C1(NC(c2[nH]cc(C#N)c2)=O)CCCC2CN(C(C3C4CC5C(C4)C35)=O)CC12 CC(O)C(F)(F)C(=O)N1CC(O)(C(C)(C)CNC(C2CC23CCOCC3)=O)C1 c1(C(=O)NC(CNC(C(C)C2CCOC2)=O)C)cnn(-c2ccccc2)c1 Cc1noc(Cl)c1CC(=O)NCC1CN(C(C2CC2(Cl)Cl)=O)CCO1 N1(C(CC(C(=O)OC)C)=O)CCC2(CC1)C(NC(C1CC(O)C1)=O)CS(=O)(=O)N2C N1(C(c2c(C(F)(F)F)oc(C)c2C)=O)CC(C)OC2(CCN(C(=O)C(F)F)CC2)C1 C#CCCCCC(=O)NC1CCC(NC(C2(CC(C)C)CCNC2=O)=O)C1 C12(SCCCS1)CCNC2=O.n1(C(C)C)cc(CC(C2CCOC2)N(C)C)nn1 C(C(C)C(F)C(=O)NCCCOC1CC1)NC(C(C)=CC1CC1)=O c1(C(CNC(C=C(C)C(C)(C)C)=O)NC(=O)CN2CCOCC2)ccccc1F S(=O)(=O)(c1ccc(Br)cc1NC1CC2(CCOC2)C1)NCc1cc(C)on1 C(C(C)(C)CCNC1CC1CN(C)C)NC(c1nc(C(=O)NCC#C)sc1)=O C1(CCC(=O)N(C2CCCC2O)C)CCN(C(C2CC3CCC3C2)=O)CC1 N1(CCOC)CCC(CC(=O)NC(C)CC(C)NC(=O)CNS(C)(=O)=O)C1 C1(CC(N2CC(C(C)(C)O)C2)=O)CCCN(C(=O)CCN=[N+]=[N-])CC1 c1(C(=O)NCC2(NC(c3ncc(C4CC4)cc3F)=O)CC2)ncn2c1CCCC2 C1(C(F)(F)F)CC2(CC(NCc3noc(-c4cccc(Cl)c4)n3)C2)C1 C(=O)(CC(O)C(C)(C)C)N1CC(C(N2CCCC(OCCC)C2)=O)(CC)C1 Cc1ccnnc1C(=O)NCC1CCN1C(c1cc(-c2ccn(C)n2)on1)=O C1(C(N2CCOCC(CNC(C3(F)CC3)=O)C2)=O)COC2COCC2O1 N1(C(C(n2cc(-c3cnc(C)n3C)nn2)C)=O)Cc2ccccc2C1 C1(CC(=O)NC23CC(NC(=O)CSCCC(C4CC4)C4CC4)(C2)C3)OCCCO1 CCCC(C(=O)NC1CCCC1NC(=O)CCCC1CCOCC1)OCC C1(NC(C)=O)CCN(C(=O)CN(CC(C)C)CC)C12CC2.c1(C2N(N)CCOC2)ccc(C)cc1C N1(C(CCCN(CCC)CCC)=O)CC2CC1C2CNC(C1OCCOC1C)=O C(C(C)N=c1cccc(S(=O)(=O)N2C3CCC2CC(CO)C3)[nH]1)S.C(CNC)OC CC1(C(=O)NCC2(O)CN(C(=O)CC3CNC(=O)C3)C2)CCOC1 Cc1noc(CCC(=O)NCCCCC2CN(C(=O)C(C)n3cnnn3)C2)n1 N1(C(CC2C(C)CCC2)=O)CCCC2(CC(NC(C3CCC=CCC3)=O)C2)C1 N1(C(CC(=O)NCC)=O)CCC(C)(CC(N2CC(c3ccncc3)C2)=O)C1 C1(C(N2CCC(C)(CNC(C3C4COCC34)=O)C2)=O)CC(c2ccccc2)=NO1 C1(NC(C2(NC(=O)CCCCC)CCCCC2)=O)CCC12CCCC2 C(=O)(C1CCc2ccc(C)cc21)NC1CN(C(CCC)=O)CC2C1C2 C1(C(=O)NCC(N2CCN(C(CC(C)CF)=O)CC2)=O)CCC2(CCOCC2)C1 c1(N2CCN(C)C(NC(=O)Cc3ccnc(F)c3)C2)nc2cc(F)ccc2o1 N1(C(CC(C)CCl)=O)CCN(CC(F)(F)F)CCNC(=O)C1 C(C(=O)NNc1cccc(Br)c1)Sc1nnc(C(=O)OCC)s1 N1(C(c2cc3oc(F)cc3[nH]2)=O)CCn2c(C(C3CCCC3)=O)nnc2C1 c1(C(=O)NCC2CN(Cc3c(OC)ccc(C)c3)C2)ccc2sc(C)nc2c1 C1(C(=O)NCCOCC(C)C)CC12CC(NC(C1(C)CC1C)=O)C2 Cc1ccncc1NC1(c2nnnn2CCC2(C)CC2)CCCC1C CCCC(C(=O)NC(C1CCCCN1C(C1(C(=O)OC)CC1)=O)C)OC c1(C(=O)OC)nc(N2CCOCC(NC(C3CC3(C)C(C)C)=O)C2)ncc1Cl CC1OC(C)C(C(=O)NCCN(C(C)(C)C)C(C2CCC(C)C2)=O)C1C CC(F)(F)CCCC(=O)NC1CCCC12CN(C(C1CCC3(CCC3)CC1)=O)C2 CC1Oc2ccccc2OC1C(=O)NCC#CCNC(=O)CCOCC(F)F C(CC(C)(C)NC(=O)CC1(C(F)(F)F)CC1)NC(C1C(COC)(CO)C1)=O C(=O)(C(CO)C(F)(F)F)NC1(C)CC(NC(C2CC(OC(C)=O)C2)=O)C1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CCC2CC1CN2C(C1CC1C(C)O)=O CCC(O)C(C)(C)C(=O)NCCN(C(C1CCCN(c2ncccn2)C1)=O)CC C1(c2ccc(C)cc2Cl)NC(=O)N(C(=O)CC(C)(C)C)C2=C1C(=O)NC2(C)C CCCC(CCC)=CC(=O)NC1CC(C)N(C(C2(NC(=O)NC)CC2)=O)C1 N1(C(CC2(NC(C3(C(=C)F)CCC3)=O)CCCC2)=O)CC2CCCC(O)C2C1 N1(C(c2c(CC)c[nH]n2)=O)CCN(C(c2cnc(C(C)(C)C)o2)=O)C(C(C)C)C1 c1(CC(=O)NCC(C)(CO)NC(=O)CCC=CBr)cccc2ccccc12 C(=O)(CCN=c1ccc(C)c[nH]1)NCC=CCNC(c1cccc(OC)c1)=O CCCC(C(=O)NC1(c2cn(CCOC(C)C)nn2)CC(F)(F)C1)C(C)C C1(C(=O)NC(CC)CNC(=O)C=C(Cl)Cl)CCCC12CCOCC2 c1(CNC(c2n(CCSC)nnn2)c2ncc(SC)s2)c(F)c(F)cc(F)c1F C1(C(N2C3C(NC(c4cc(CC)ncc4)=O)C(C3)C2)=O)CCC=CCCC1 c1(CNC(C2N(C(C(CSC)O)=O)CC=C2)=O)cccc(F)c1F c1(N(C(=O)CN2CC=CC2)C)ccc(CCCNC(=O)OCCl)cc1.C(C)(C)(C)O S(=O)(=O)(CCCCS(N)(=O)=O)NC(=O)NCCCOc1cc(C)cc(F)c1 N1(C(C(CSC)(C)C)=O)CCC(C2CC2)C1C(=O)N(C)Cc1ccon1 C=CC(CCC)CC(=O)NCC1(C)CCN(C(=O)C(C)NC(C2CCCC2)=O)C1 C(=O)(C1=NOC2(CCOC2)C1)NCCC1N(C(C(C2CCC2)OC)=O)CCSC1 C(C)(N=c1ccnc(NCc2ccc(Br)s2)[nH]1)c1c(OC)ccnc1O c1(C(=O)NCC2N(C(CC=CCC)=O)CC2)cnc(C(C)(F)F)s1 C1(OC2CN(C(C(C)C3CC3)=O)C2)CCN(C(=O)C(F)CC2CCCCC2)CC1 c1(C(=O)NCCC(C)N(c2ncnc(C)c2F)C)cc2nn[nH]c2cc1F C1(C(=O)NOCCF)(NC(c2coc(C3CCCC3)c2)=O)CC(F)(F)C1 c1(OC2(CC(=O)NCC(C)CNC(C)=O)CC2)ccccc1 c1(C(N2CC(NC(c3n(CC)nc(C)c3)=O)C(C)(C)C2)=O)cccc2c1OCO2 C1(C(=O)NC2C3CCN(C(CCc4c(C)n(C)nc4)=O)C32)CC(C)(C)OC1(C)C C1(NC(COCCCC)=O)CN(C(c2ncccc2O)=O)CC1SC C(=O)(C(F)C(F)(F)F)NC1CC(F)(CNC(c2ccccc2OCCF)=O)C1 C(=O)(C1=CCCCC1C)N1CC(C(C)(C)O)(CNC(CCC=CC(C)C)=O)C1 c1(Nc2c(Br)cnc(SCCC)n2)cc(OC)c(Cl)cc1OC S(=O)(=O)(c1cccc(I)c1)NC(c1n(C)c2c(n1)CCCC2)=O CCCC(CC)C(=O)N(C(CC(F)F)C(=O)N1CC1)C.C1(OC)CC1 C1(C(=O)NCC(CCC)O)CN(C(=O)C(c2cccn2C)=O)C2(CCC2)C1 c1(C(=O)OC)cccc(C(N2CCSCC2c2nccs2)C(=O)NC2CCC2)n1 C1(NC(C(C)SCCCC)=O)CC2CCC1N2C(c1nccc(C)n1)=O CC1CC(NC(C2CCOCC2(C)C)=O)CN(C(=O)C=CCO)C1 c1(C(c2nn(C)cc2Cl)NC(=O)NC2C(C)C2C)cc(F)c(Br)cc1F C1(NC(C=CCN(C(=O)CC2CC(F)(F)C2)C)=O)CCC(N(C)C2CC2)CC1 C(=O)(CC1=CCN(C)CC1)NC(CC(C)C)(C)CNC(=O)C(F)C(C)(C)O C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1OCC(CNC(C2CCC(SC)CC2)=O)C1 c1(OC)c(C(=O)NC2CC3CN(c4ncc(C)c(SC)n4)CC3C2)cc(F)cc1F N1(C(C(=O)NCc2c(OC)nccc2)=O)CCC2OCCNC2C1 CC(C)CC(CNC(=O)COCC1CCOC1)C(=O)N1CC2C(C)C2C1 C1(CC#N)CN(CC2CC2(F)F)CCN1C(=O)Cc1ccc(CC#N)cc1 C1(NC(=O)CCCN2CCCCC2)C2CN(C(=O)C(F)CC3CC3)CC12 c1(NCCOCC)cccc(F)n1.c1(C(CC)(C2CC2)N)nnnn1-c1ccccc1 C=CC(C)(C)CC(=O)N1CC(CNC(c2cnc(O)c(C)c2)=O)C(C)C1 N1(C(C=C(CC)CC)=O)CC2CCCC(C1)N2C(c1cc(Cl)n[nH]1)=O CC1CN(C(C2(F)CCOC2)=O)CC(C)N(C(=O)COc2cc(F)ccc2F)C1 N1(C2N(C(=O)CCCc3sccc3C)CC(NC(C(COC)C)=O)C2)CCC(C)(C)C1 c1(C(=O)NCCN(CC(C)O)C(=O)CC2CCCC(=O)N2)cnc(O)n1C N1(C(C2COCC(C)O2)=O)CCC2(CC2C(=O)NCCc2ncc[nH]2)C1 c1(C(=O)NC(C)CN(C)C)ccc(S(=O)(=O)CC(C)(C)C)cc1 C(=O)(CCS(C)=O)N(C(C)C)CCN(C)C(c1cccc(NC2CCCC2)c1)=O C1(CN(C)C(c2coc(Br)c2)=O)CN(C(=O)Cc2cn[nH]c2)CC12CC2 C(=O)(C(CNC(c1nnc(S)n1C)=O)(CC)CC)NC(CCSCC)C c1(C(N2CCN(C(c3ccccc3[N+](=O)[O-])=O)C3CC23)=O)cc(F)ccc1Br N1(C(C2(C(=O)NC)CCC2)=O)CC=CC1CNC(C1CC1C(C)(F)F)=O C1(C(=O)NCC2CCCC(NC(C3CN(S(C)(=O)=O)C3)=O)C2)CC1C1CC(F)(F)C1 c1(C(=O)NCCNC(c2cccc3nsnc23)=O)cc([N+](=O)[O-])c2nsnc2c1 c1(C(N2CCN3CCCC3C2)=O)cccc(S(=O)(=O)NCC2CCC(F)(F)C2)c1 c1(C2CC(CNC(=O)NC(C)Cn3cncn3)C2)cccc(F)c1 CC(C)CCCCNC(=O)C(C1CC1)N(C(=O)C(C)c1cccs1)C N1(C(C(c2ccccc2)C)=O)CCCN(C(=O)NCCC(=O)O)CC1 CC1(C)CC(CNC(c2cc(Cl)nn2-c2nc[nH]n2)=O)N(C(C2CCSC2)=O)C1 C1(C(=O)NC(C2CCN(C(=O)C=Cc3cccs3)CC2)C)CCn2nncc2C1 CCC(C(F)(F)F)NC(C1CCCC1NC(c1c[nH]c(=NC)o1)=O)=O N1(C(COC(C)=O)=O)CCCC2(CCN(C(c3ccnc(CC(C)C)n3)=O)C2)C1 C1(C)(C(=O)OC(C)C(=O)Nc2ccccc2C(F)(F)F)CC2CC2C1 CC1CC(NC(C2CC(C#N)C2)=O)CCN1C(=O)Cn1nnc(-c2cccs2)n1 c1(CCC(=O)N(C)Cc2ccc(CC)c(F)c2)ccc(Br)cc1F N1(C(c2cccn3nccc23)=O)CCCC(C2CCN(c3nccnc3F)C2)C1 CC1CCC(CNC(C2CCC(SC(C)C)C2)=O)O1.C12(CC1)C(=O)N2 N1(C(c2ccn(C)c2)=O)CC2(CCN(C(C3C4C(=O)OCC34Br)=O)C2)C1 N1(C(C(C)(C)O)=O)CC2C3CCC(C(NC(c4ccc(F)c(CO)c4)=O)C3)C2C1 Cc1cnc(NC(c2c(F)cccc2F)(C)C)nc1C c1(COC)cc[nH]c1C(N1CC(C)C1C(=O)NCCCSC(F)F)=O C(=O)(CC(C)CC(=O)NC1CCC(CNC(=O)C(C)N(C)C)C1)OC C1(C(N2CC3(CCN(C(=O)C(Cl)=CCl)C3)C2)=O)CCOCC12CCCCC2 c1(C(=O)OCC)cc(Cl)cc([N+](=O)[O-])c1NC(=O)CCCSC Cn1nnc2c1CC(C(=O)NCC1CCCC1NC(=O)CC=C(Cl)Cl)CC2 N1(C(C23CCC(OC)(CC2)C3)=O)CCN(C(=O)C(C)O)C2CCCCC12 N1(C(C2N(C(CNC(CC3C(C)(C)C3)=O)=O)CC2)=O)CC(C)(O)C1 N1(C(C)=O)CCCC(C(=O)NC(CNC(c2ccc(F)cn2)C2CCCC2)C)C1 Cc1conc1S(=O)(=O)Nc1ccc(C2(C)CCO2)cc1 C(=O)(CC(F)(F)C(F)F)NCC1CCCN(C(c2c(OC)nc(Cl)cc2)=O)CC1 N1(C(CCN2C(=O)CCCC2=O)=O)CCC2CC1CN2C(=O)C=CC1CCC1 N1(C(c2c(F)ccc(C)c2)=O)CCC2CC2(NC(c2ccc(F)s2)=O)CC1 c1(OC)ccc(C)nc1C(=O)NC1CCCC(NC(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(=O)NC2(C)CN(C(C3CC(OC)C3)=O)C2)cn(CCO)nc1C C1(C(=O)NC2CC(CNC(CC(C)(C)SC)=O)C(O)C2)CCn2c(C)nnc2C1 N1(C(C(N)=O)=O)CCCC(F)(C(C2CC2)NC(=O)CC2(CSC)CC2)C1 N1(C(C(C)C)=O)CCC2(COC(CNC(C3C(C)(C)C3(C)C)=O)C2)C1 c1(CCC(=O)NCC(CC)NC(C2(CC#C)CCCC2)=O)ccccc1Cl Cc1nc(C(N2CC3(NC(=O)CCC4CC4)CCC2C3)=O)c(C)n1C N1(C(C(c2ccccc2)OC)=O)CC(C2CCCN(C(C3CC(C)(C)C3)=O)C2)C1 C12(CC(=O)Nc3c(COC)n(C)nc3)CCC1CN(C(=O)CN=[N+]=[N-])C2 Cc1nc2cc(Cl)c(NC(C3CCC(NC(=O)CCC(N)=O)C3)=O)cc2o1 N1(CC(=O)N)C(=O)C2C3CCC(O3)C2C1=O.N1(C)CCC(c2nc(C(=O)O)n[nH]2)CC1 S(=O)(=O)(c1nccs1)NC1CCC(Nc2c(OCC=C)cccc2)CC1O N1(C(c2scc(C#N)c2)=O)CC(NC(C2CC2F)=O)CC12CCOCC2 C12(CNC(c3c(CC)ncs3)=O)CN(C(C3(C)CC(F)C3)=O)CC1CCO2 N1(C(C(CC)c2ccccc2)=O)CC(c2ccccc2)C(O)C1 n1(CC(=O)NCCSCC(=O)NC(CCSC)C)nc(C)nc1C Cc1ccc(C(N2CCC(N(C)C(c3cccn3C(C)C)=O)CC2)=O)c(F)c1 C(CC(C(C)(C)C)NC(=O)Cc1nnc(S)n1C)N(C(C1C(=C)CC1)=O)C C#Cc1ccccc1CC(=O)NC(C1CCCN1C(=O)CCC(C)(F)F)(C)C C1(NC(c2cc(CCC)on2)=O)CN(C(c2cn(C)nc2O)=O)CCC1O c1(OC)nc(C)cnc1-c1nc(-c2cc(C)cc(C)c2)no1 Cc1oc(Br)cc1C(=O)N(C)CCOCCCNC(=O)C(C)(F)F CCC(CC(C)C)C(=O)N(C)CCNC(C1CNC(=O)C(C)(C)C1)=O N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CCC(NC(=O)CCS(C)=O)C2(CCC2)C1 c1(COC(N2CCCC(C(C)NCC(F)(F)F)C2)=O)cc(Cl)c2c(c1)OCCO2 CC1Oc2ccc(C(=O)N(CCCNC(c3cnc(Cl)s3)=O)C)cc2C1C C(=O)(C(C(C)NC(c1cnc(C)cc1C)=O)C(C)C)N(CC(=O)NCC)C O=C(CN=c1cc[nH]cc1)N1CC(SCCNC(=O)COC(F)(F)F)C1 N1(C(c2c(CNC(C(c3cnn(C)c3)C)=O)nccc2)=O)CCCC12CCCC2 N1(C(C2(CC=C)CC2)=O)CC(NC(C2CC(N(C)C)C2)=O)C(C)(C)C1 N1(C(=O)OC)CC(NC23CCCC(C(=O)OCC)(C2)C3)C2(CCC2)C1 Cc1cc(C(O)CN(C2CC2)Cc2ccc(OC(F)F)cc2)ccc1F c1(CC(NOCC(C)(C)C)=O)cnc(Cl)cc1Cl c1(C(=O)NC2CC(C(C)NC(c3ccc(CCC)s3)=O)C2)cccc2ccoc12 C1(c2n(CCCC)nnn2)(NC(c2cc(F)ccc2C)CC)CCN(CC)CC1 c1(C(C)C)cc(C(=O)N(CC(C)(C)NC(=O)COCCOCCO)C)on1 C1(NC(C2C(C)(C)OCC2)=O)CCN(C(=O)COC2CCCOC2)CC(O)C1 CC(C)C(C(=O)N(C1CCCN(C(=O)CC(F)(F)Cl)C1)C)N1CCCC1 O=C1CN=C2C=CN=C(N2)N1.c1(NCC2CCC3CC23)nc2ccccc2s1 N1(C(C2CC2c2ccc(F)cc2)=O)CCOC(c2cn(NCC3CCOC3)nn2)C1 N1(C(C(CCNC(c2ncnc(C)c2C)=O)O)=O)CCc2cc(C#N)ccc21 C1(NC(C2CC(C#N)C2)=O)CN(C(C2CCOC2C2CC2)=O)C2(CCCCC2)C1 C=C(C)C1OCCC1C(=O)N(CCCCCCNC(=O)CCSCCCC)C c1(CC)ncncc1C(=O)NC1CC(F)(CNC(c2ccnc(C(F)F)c2)=O)C1 N1(C(C(=O)Nc2cccc(OC)c2)C2CC2(C)C)CCC(O)C(C)C1 N1(C(CCCOC(C)=O)=O)CCn2ncc(CNC(=O)Cc3ccon3)c2C1 c1(CCNC(C2C(C(=O)Nc3c(C#N)cns3)C2)=O)cc(F)cc(F)c1 C1(NC(CCC2(C)CC2)=O)CC2CC(C1)N(C(=O)C=Cc1cocn1)C2 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCCOC2CCOC2)C1 Cc1nc[nH]c(=NCC23CCCC2CN(C(=O)C=C2CCC2)C3)c1Br n1(NC(=O)O)cc(CC(C(=O)OC)NCC(C)(C2CC2)NC(C)=O)nn1.C(C)(C)(C)OC C(=O)(C(CC(C)C)C(C)C)NC(CC#C)(C)C(=O)Nc1cc(COC)ccc1C c1(C(=O)OC)cc(F)c(C)c(NC(c2nccc(C)c2N)=O)c1F c1(C)ccc(C(=O)ON2CC(C)(CC(N3CCCC3C(N)=O)=O)C2)cc1.C(N)=O N1(C(c2c(CC)[nH]nc2Cl)=O)CCN(C(=O)C(=Cc2cccnc2)F)C(C)C1 C1(c2cccc(C(=O)OCC)c2)CCN(N2CCCN(CC)CC2)CC1 c1(C(=O)OC)ccc(C2(C(=O)Nc3nccc(Oc4ccccc4)n3)CC2)cc1Cl N1(C(C2C(COC)CC2)=O)CCSCC1C(=O)N(C1COCC1O)C N1(C(=O)Nc2ccnn2C(F)F)CCC(O)(C(N2CCCCC2CO)=O)CC1 C12(CNC(C3CC(CCC)C3)=O)CCCC1CN(C(=O)C(C(CC)CC)OC)C2 NC(=O)CCCC(=O)NCCN1CCN(C(c2cn(CCF)nn2)=O)CC1 CCC(CC(=O)NCC(=O)NCC)OC.C1CC(=O)NCCO1.C(C)=O c1(CNC(=O)NC(CC(=O)NC)C)cc(C#N)ccc1Br O=C(CC1C(=O)Nc2ccccc21)NC1(O)CC(CNC(=O)COC(F)F)C1 N1(C(CC2C(=O)OCC2)=O)CC23CCCC2(C1)CN(C(c1c[nH]nc1Cl)=O)C3 c1(C(=O)NC2CC3(C2)CN(C(C2CCCC2O)=O)C3)cc2c(Cl)cc(F)cc2[nH]1 C1(NC(C2(C#C)CC2)=O)CCC2CN(c3nc(C)nc4sccc34)CC2C1 n1(CCOC)cc(C(=O)NCCC2CN(C(C)=O)CC(C)O2)ccc1=O CC(C)C(O)CC(=O)NC(C1(O)CN(C(=O)CC2(c3ccon3)CC2)C1)C Cc1cc(C)c(C(=O)N(C)CC2COCCN2C(C2CC2CN(C)C)=O)cc1C c1(C(=O)NCC(C)CN(C)C(C2(C)CC=CCO2)=O)ccc(-n2cnnn2)cc1 c1(C(=O)NC2CN(C(c3c(CC)n(C)nn3)=O)CC2(C)C)cc2n(n1)CC(F)C2 N1(C(c2cnc(C)n2C)=O)CCC(C(=O)NC(CO)C2(C)CC2)=C(F)C1 N1(C(c2c(Cl)ccc(NC(C)=O)c2)=O)CCC(C)C(NC(=O)C(N)=O)C1C C(=O)(CCCC(C)=O)N1CCN(C(=O)C2CC2)CC1.C#CC12CN(C1)OC2=O Cc1cc(F)cc(C(N2CC(NC(C34CCCN(CC3)C4)=O)C2)=O)c1N C1(C(=O)NCCN(C(=O)COc2ccc(Cl)cc2F)CCC)CN2CCN1CC2 CC1(C)CN(C(=O)CC2(O)CC2)CCC1NC(C1COCCO1)=O C(c1cccc(O)c1)=CC(N1C(C)CC(CNC(Cc2cc(C)sc2)=O)C1)=O C1(NC(C(C=C)O)=O)CN(C(C2CCCC23CCC3)=O)CC2(CC2)C1 CC1CCNCCC1N(C(C1CCC(=O)NC1)=O)CC1CCOCC1 C(=O)(CCCC(=O)NC(C1CCCC1)CNC(C1(C)CC(C)=NO1)=O)OCC c1(C(=O)OC)ccc(C(=O)NC2CC(C)(NC(C3C=CCCC3)=O)C2)n1C CC12CC(C(=O)NC3CC3NC(c3cnoc3-c3cccs3)=O)(C1)C2 c1(C(C(N2CCN(CCNC(C3(Cl)CC3)=O)CC2)=O)O)ccc(F)cc1 N1(C(C2(CNC(CC(COC)C)=O)CCCC2)=O)CCNC(=O)CC1C C1(CC(N2CCC(NC(CC)=O)C(O)C2)=O)Cc2cc(Br)ccc2C1=O N1(C(C2N(CCC)CCC2)=O)CCC=CC1C(=O)N(C)Cc1ncnn1C C1(C(=O)NCC(CCC)NC(C(CC(=C)C)NC(C)=O)=O)CCn2cncc2C1 N1(C(c2ccc(C)s2)=O)CCC(NC(=O)CNC(c2ccc(Cl)cc2)=O)C(F)C1 CC1CCCC(C(=O)NC2CN(C(=O)CCc3ccsc3)C2)CC1 C1(C(=O)NCC(CNC(c2nc(C(C)(C)C)sc2)=O)O)CCCC2C1C2(F)F c1(C(=O)NCC(CC)NC(=O)Cc2c[nH]nc2O)nc(Cl)sc1Br CC1(C)CC(CNC(=O)CSC(F)F)N(C(C23CCC(F)C2CC3)=O)C1 C(=O)(CN=c1[nH]c2c(c(=NCC3CCC(O)C3)[nH]1)CCC2)NCC=C c1(C(=O)NCC2OCCN(c3nccc(C(=O)OC)n3)C2)noc2c1COCC2 C(=O)(CS(=O)(=O)CC1CCCO1)N1C(C)C(NC(=O)C=CCN2CCC2)CC1 C1(OC)CCC(C(N2CCCC(N(C(=O)CSc3nc[nH]n3)CCF)C2)=O)CC1 C1(C(N(C)CC2CN(C(=O)CC3CCC3)CCO2)=O)CCN(CCO)C(=O)C1 CC1OCCC1(F)C(=O)NCc1cc(C(=O)NCC2=CCSC2)ccn1 N1(C(c2c(C)scc2)C(=O)NCc2ccccc2)CCCC(C#N)C1 N1(Cc2n(C(=O)OCC)c(O)nn2)C(CO)CC2CCCC12.C1CO1 CC1(C)CC2(CCC2)CN1C(=O)CCN(C(c1cc(O)cs1)=O)C1CC1 Cc1cc(C(=O)OC(=O)C(c2cscn2)NC(=O)OC(C)(C)C)c(Br)cc1F c1(CC(=O)NCCNC(C2(C(C)C)CCC2)=O)cccc(N2CCOCC2)c1 N1(C(C(CCC)CC)=O)CCc2[nH]nc(CNC(C3(C4CC4)CC3)=O)c2C1 c1(C(N2C3C(N(C(c4c(C)nccn4)=O)C)CC(C3)C2)=O)cc2c(nn1)CCC2 N1(C(c2ccc(C)cc2Br)=O)CC(NC(C2CC(O)C2)=O)CC2(CCC2)C1 C12(C(=O)NC3(C)CN(C(c4cnc[nH]c4=N)=O)C3)CC3CC1C2C3 Cc1cc(=NCC#CCCO)[nH]cc1S(=O)(=O)N1CCC(NC2CC2)CC1 c1(NC(C(COC)N(C)C)=O)n[nH]c2c1CN(C(=O)C(O)P(C)(C)=O)C2 C(C)(C(O)C(=O)NCC1(F)CC(CNC(c2ccccc2Cl)=O)C1)SC CC(C)(C(=O)NCC1CN(C(=O)CCc2ccco2)C1)C(F)c1ccccc1 C1(NC(c2c(CC)ncs2)=O)CCCCN(C(c2ccccc2C(=O)NC)=O)C1 [N-]=[N+]=NCC(F)CCNC(C1CC(NC(C2CCCCCCC2)=O)C(O)C1)=O C1(NC(C(C)NC(=O)NC)=O)CC2CCC1C(NC(=O)C(F)(F)CO)C2 C1(C)(C(N(C(C)C)CCNC(C2C(C)C2C)=O)=O)CC2(CCC2)C1 N1(C(C(C)NC(=O)C(C)C(=O)NC(=O)C(C)C)=O)CCCC(F)CC1 Cc1ncc2n1CCN(C(=O)C(C)C(C)NC(=O)C(C)c1ccco1)C2 CC(C)(CNC(C1CCOC(=O)CC1)=O)CC(=O)NCC1CC(O)C1 C12(C(N)=O)CC1CN(C(C1CCC(=O)N1C1CCCC1)=O)C2 c1(C(N2C3CC(NC(CCCCCC#C)=O)(C3)C2)=O)cc2n(c1)CCS(=O)(=O)C2 N1(C(C2CC(O)C2)=O)CC2(C1)CN(C(=O)C1=CCCCO1)C2 c1(C(N2CCC(N(CCC)C(C3CN(C)CCO3)=O)C2)=O)ccc2c[nH]nc2n1 C(=O)(C1=Cc2ccccc2OC1)NC1C(C)CCN(C(=O)CC2CCOC2=O)C1 C(c1ccc(F)cc1)=CCC(=O)NCC1CN(C(c2c[nH]c(=O)cn2)=O)C2CC12 c12ocnc1C(=O)NC2.CC(C)(C)CC1CCN1C(=O)C=CC(F)F C1(NC(CNC(C)=O)=O)CCCCC12CCCN(C(c1ccc(=N)[nH]c1)=O)C2 C(CN=c1nc(-n2cccn2)cc[nH]1)C1CCN(c2sccc2)CC1 C1(F)(C(=O)NC(CCOC)CNC(c2cc(C)cs2)=O)CS(=O)(=O)CC12CCC2 N1(C(c2ccc(COC)cc2)=O)CC(CO)C2(C1)CN(C(c1coc(Br)c1)=O)C2 C1(C)(C(N2CCC(C(C)C(=O)NCc3cnsc3)C2)=O)CCOCC1 c1(C(N2C(CN(C(C3C(C=C)OCC3)=O)C)COCC2)=O)cc(N)c(C)cc1C N1(C(c2[nH]cc(C(N)=O)c2)=O)CCN(C(=O)Cc2ccon2)CC1 C1(C(=O)NC(c2cn(CC)nc2)C)CN(C(=O)C(O)C(F)(F)F)CCN1C Cc1nc(S(=O)(=O)N2CCCCC2C(N2CSCC2C(=O)O)=O)cn1C c1(C(=O)NCc2ccc(C)cc2F)n[nH]c2c1CN(C(=O)CC1CCC(O)C1)C2 c1(CC(=O)NCCN(C)C(C2CC3C=CC2C32CC2)=O)ccc2[nH]ccc2c1 C(C(C(C)C(C)C)NC(c1nc(O)c(C)s1)=O)NC(COCCCCCC)=O c1(SCC(=O)NC2C(NC(CCCSCC=C)=O)CCC2)nnc(COC)n1C C1(N(C(c2coc(C(F)F)c2)=O)CC)CCCN(C(=O)CCOCC(F)(F)F)C1 c1(CC)nccnc1CNC(=O)CC1CC1CNC(C12CSCC1C2)=O c1(CC(N2CC(c3cn(-c4ccccn4)nn3)C2)=O)nnc(S)n1CCCF N(C(=NCC1C(C(=O)OC(C)(C)C)C1)NCC(C(C)(C)C)SCC#N)C(C)C N1(C(C(C(C)(C)C)NC(C(n2c(C)ncc2)C)=O)=O)CCC(C2CCCC2)C1 C1(CC(=O)NC(CC2CC2)C2CC2)CC(N=c2ccnc(C(F)(F)F)[nH]2)C1 N1(C(C2(CO)C(C)C2)=O)CCC2(CCC(NC(=O)C3=NNC(=O)CC3)CC2)C1 C(C(=O)NC(C)CNC(=O)C(c1cc(C(F)(F)F)c[nH]1)=O)(C(C)C)OCC(C)C n1(C(C)C(=O)NCC2CC(CNC(C3(C(F)(F)F)CCO3)=O)C2)cc(Cl)cn1 Cc1cc(CC2CC(NC(=O)C=CC(=O)Sc3ccccc3F)C2)cc(F)c1F c1(CC#N)ccsc1C(=O)NCCC(Cc1ccccc1)NC(C1CCCS1)=O C(=O)(C(C)CC)NCC(=O)N(CCNC(C1CC(=C)C1)=O)CCOC C(=O)(CC(C(C)OC)NC(C1CC(C)(C)CO1)=O)NC(C=C)COC N1(C(=O)NC2(CCO)CCCO2)CC(C2CC2)(CNC(=O)OC(C)(C)C)C1 N1(C(=O)NC(COC)C)CCC(NC)CC1.c12cccc(c1)CN2 N1(C(C2CC2C2CC2)=O)CCC(F)(CNC(C2(c3ccc(F)cc3)CCC2)=O)C1 C1(C(N2CC(C(CC)C)C2)=O)C2CCC(C2)N1C(C1(CO)CCCO1)=O c1(CC(=O)NCC2CCCCN2C(c2ccc(F)c(O)c2)=O)ccnc(F)c1F C=CCCCCCC(=O)N1CC(C)(NC(=O)CN(C)S(N)(=O)=O)C1 Cc1ccc2c(c1)OC(C)CN2C(C1CCCCC1)C(=O)NC1CCS(=O)(=O)C1 C1(CCC)(NC(COCC=C)=O)CCCN(C(C2CC23CCCCC3)=O)C1 N1(C(C(CC)=CC)=O)CC(NC(c2cccnc2Sc2ccccc2)=O)C(C)C1 C(CC(=O)NC(C1CC(F)(F)C1)C)(C(C)CC)NC(c1nccc(C#C)c1)=O N1(C(C(C)N(C)C)=O)CCC(C2CCN(C(c3ccc(N)c(SC)c3)=O)C2)CC1 N1(C(CN2CCN(C(CC(C)N(CCC)C)=O)CC2)=O)CCC(F)(C#N)C1 CC(C)(CC(F)C(=O)NCCc1nc[nH]n1)NC(C1CC12CC2)=O N1(C(c2c(CC)ccs2)=O)CCC(C)CC1CNC(=O)CC1(CO)CC1 N1(C(C2(NC(CCCOC(C)(C)C)=O)CSC2)=O)CCCCC(F)(F)C1 C#Cc1ccc(CC(N2CCC(C(C)NC(=O)C(C)C(F)(F)F)CC2)=O)c(F)c1 C(=O)(C1=CCN(C(=O)C(C)C(F)(F)F)CC1)NC(CC)CC C1(CNC(=O)CC2CCCO2)CC2(CCN(C(=O)CNC(=O)CNC=O)C2)CO1 c1(C(N2CC(C)C(NC(C3(C)CCCC3C)=O)C2)=O)n[nH]c2cccnc12 N1(C(C(C)(C)OC)=O)CC2CCCC(NC(c3coc(O)n3)=O)C2C1 N1(C(CC2CC(C)(C)CN2C(=O)CCCF)=O)CCCC2OCCC12 N1(C(c2c(C)ccs2)=O)CC2CCC2(NC(c2ccc(C#N)[nH]2)=O)C1 C#CCC(CC(=O)OC)N(C1CC1)CC1(C)CCCC(=O)N1 c1(CN2CCN(C(=O)NC3CCCC3)CC2)cc2ccc(F)cc2nc1O N1(C(CCCC#C)=O)CC2(C(N3CCCC(CC)CC3)=O)CC1CO2 CCC(C)C(C(=O)N(C1CCN(C(=O)CCC2CCCC2)C1)CC1CC1)SC c1(C(N2CCC3CCC(C2)N3C(C2(F)CC2(Cl)Cl)=O)=O)ccc2c(c1)NC(=O)C2 N1(C(C(N2C(C)C(c3ccccc3)CC2)=O)=O)CC2C3CCC(C3)C2C1 c1(CC(=O)NC2CC(CNC(C(C3COC(C)(C)O3)O)=O)C2)c(F)cccc1Cl Cc1cc(S(N)(=O)=O)oc1C(=O)NC1CC2CC(NC(=O)CC(C)C)CC12 c1(C(=O)OC)ccc(=NCC2CCN2CC(=O)NC2CCC2(C)C)[nH]c1C C1(NC(=O)CCF)CC(F)CN(C(C2CCN(Cc3ccccc3)C2=O)=O)C1 C1(CC(=O)OCC)CN(S(=O)(=O)c2ccccc2C(C)C)C2(CCC2)CO1 C1(C(=O)NC2CCC(N(C(=O)CSC(F)F)C)CC2)C(C2CC2)C1(F)F C1(C(=O)Nc2nc(C)sc2)C(C2CC2)CCN1C(=O)CCc1ccn(C)n1 C1(C(N2CC3CN(c4ncc(I)cn4)CC3C2)=O)COc2ccccc2O1 N1(C(c2nc[nH]n2)=O)CCN(C(C2(c3ccccc3)CCCCO2)=O)CC1 N1(C(C=Cc2n(CC)ncc2)=O)CCCC(NC(=O)CSC(F)F)CC1 C=C(CNC(C12CCC(C1)C2)=O)CCNC(c1coc(C)n1)=O C(c1ccnn1C)=CC(=O)N(C1CCN(C(c2cccnc2S)=O)C1)C Cc1cc(C(=O)N(CC(CO)(CO)NC(=O)C(C)OCC(F)(F)F)C)ncn1 Cc1ccc(C=CC(=O)NC2CC(CCC(=O)NC(C3CCOCC3)(C)C)C2)o1 c1(OC)c(F)ccc2c(C(=O)NCc3ccc(Cn4cccn4)cc3)[nH]nc12 c1(C(=O)NC2C(CC)CN(C(C3CCSC3)=O)C2)cc(C)nc2ccccc12 N1(C(C(C)S(N)(=O)=O)=O)CCN(c2nc(C3CC3)nc(=N)[nH]2)CC(O)C1 N1(C(C(C)Cc2ccccn2)=O)CCC(C)(CNC(=O)C(F)C2CCOC2)CC1 CCC(C)C(=O)NCC1(CCNC(=O)CC2CCCSC2)CC1 C1(F)(C(=O)NC(CC=C)CNC(C2CCCN(C(=O)NC)C2)=O)CCCCCC1 C(C1=NOC2CN(C(c3coc(C4CC4)n3)=O)CC12)NC(C(CC)(C)CC)=O C1(C(=O)NCCC(C)OC)CC(NC(c2ccsc2OC)=O)C(O)C1 C(CCCC(=O)NCC1CN(C2CC2)CCO1)N(C)C(C1CCCN1C1CC1)=O c1(OC)ccc2c(c1)OCCC2C(=O)NC1CCC1CNC(c1ccsc1Cl)=O Nc1nonc1C(=O)NCC1(C(=O)NC2CCCC2O)CC1 C1(OC)CC(CNC(=O)CCCCn2ccnn2)N(C(=O)CSc2cccs2)C1 c1(C(=O)NC2(C)CCCN(C(C3CC(CF)C3)=O)C2)ccc(Cl)c2occc12 C(=O)(CC(C)(C)c1ccc(F)cc1)NC1C(CNC(c2c(C)noc2)=O)CC1 CCCCC(O)C(=O)N1CC(C(O)C(=O)NC2CCN(C(N)=O)CC2)C1 C1(CNC2CCCC(C(=O)OC)CC2)CC2CCC1CC2O C(=O)(C1=CSCCO1)NC1CC(NC(CN2CC(=O)NC2=O)=O)CC1O C1(C(c2c(C)[nH]c3ccccc32)=O)CCC(N=c2[nH]ccn3ccnc23)CC1 N1(C(COC)=O)CCCC(C(C)(C)C(=O)N2CC(C)(OC)C2)C1 c1(NC(C(=O)NCC23OCCC(C(=O)OC)(C2)C3)=O)n[nH]c2ccc(F)cc12 c1(OC)cnnc(OC)c1C(=O)NC(C)CNC(c1cn(C)cn1)=O c1(NC)cnc(Cl)cc1C(=O)NC1CCN(C(=O)OC(C)(C)C)C(C)C1 C(=O)(C(F)(CNC(=O)CC1CC2C=CC1C2)C(C)C)NC(c1nn[nH]n1)CC c1(C(C)NC(C(C2CCCC2)NC(C(C)=CC=C)=O)=O)snnc1C C=CC1COCCN1C(C1(NC(c2ccc(CC)nn2)=O)CC1(C)C)=O c1(CC(=O)NCC2(O)CCCN(C(CCCC#C)=O)C2)cccc([N+](=O)[O-])c1C c1(NC(N2CC(c3cccc(C(=O)OC)c3)C2)=O)ccc(Cl)c(C)c1Cl S(=O)(=O)(c1c[nH]c(=NCCc2ccc(C)s2)cc1C)NCCS(CC)=O c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CC2)ccncc1C c1(C(N2CCC(NC(c3ncn(CC)c3)=O)C2C)=O)ccn2nccc2n1 Cc1ccc(C(=O)NCC(C(C)C)NC(=O)C(C)(C)N(C)C)o1 C=CC(C)(C)CCNC(C1(CNC(=O)Cc2ccccc2C)CC12CCC2)=O c1(OCC(N2CC(N(C(C(C3CCC(=O)N3)C)=O)C)C2)=O)ccc(Br)cn1 C1(C(=O)NCCCCCN(C(C(C)(C2(C)CC2)OC)=O)C)CN(CP(C)(C)=O)C1 N1(C(c2c(Cc3cnc(CC)s3)cncc2)=O)CCC(N2CCCCC2)CC1 C(=O)(C1=NN(C)C(=O)CC1)NC12CC(CNC(CCn3ncc(C)c3)=O)(OC1)C2 C12(CNC(CCC=CC)=O)CCC(C1)N(C(c1ccc(C3CC3)cc1F)=O)C2 C1(CNC(CC2N(C(c3c(OC)csc3)=O)CCC2CC)=O)CC(C2CC2)=NO1 CC1=C(C(=O)NCC2C(C(c3cc(C)ccc3C)=O)C2)CCO1 c1(OC)cc(NC(C2CC(F)CN(C(=O)CC(C)(C)C)C2)=O)ccc1C C1(C(=O)NCC2CN(C(CC3N(CC)CCOC3)=O)C2)Cc2ccccc2CO1 C1(NC(CSCCN(C)C)=O)CCC(CCNC(c2cn[nH]c2)=O)C1 CC1(F)COCCN(C(=O)CCCCCCNC(C2CN(C(N)=O)C2)=O)C1 C1(Cn2cc(C3CCCN(C(C4(C(N)=O)CC4)=O)C3)nn2)CC(C2CCC2)C1 Cc1ccc2sc(C(=O)N(CC(O)CN(C(=O)CCOC3CC3)C)C)c(C)c2c1 c1(C(N2CC(NC(CC(=O)OC)=O)CC23CCC3)=O)cccc2c1ncn2C C1(C(=O)NCCN(C(=O)C(C)(F)F)CCC)COC2(C1)CS(=O)(=O)C2 C(=O)(CCS(N)(=O)=O)NC(C1N(C(CCCCC)=O)CCC1)C C=CCC(CC=C)C(=O)NC(CC1CC1)C(=O)NOCCF N1(CC=C(C)C)CCc2c(O)cccc2C1.C1(CC(=O)N)CCCC1C N1(C(c2n(C)c(-c3ccccc3F)cc2)=O)CCCCC(NC(=O)C=CCF)C1 CCC(C(=O)OC)n1ccc(C2(n3cc(Br)nn3)CC2)n1.CC O=C(CN1CCn2cnc(-c3cnn4c3CCC4)c2C1)N=c1ccnc(OC)[nH]1 C1(C(=O)NCC(CN(C(C(CC#C)C)=O)C)O)CC2(C1)CS(=O)(=O)C2 C1(OC)CCC2(C(=O)NCC(C)NC(=O)Cn3cccn3)CC12 C(=O)(C1=CCC(F)(F)CC1)N1C(C(=O)NCCCOCC)CCC1 CC1CN(C(=O)C(C2CC2)O)CCN1N1CCOCC1.c1(C=O)nc(Cl)ncc1Cl C(=O)(C(C)(CNC(=O)CN(C)S(N)(=O)=O)CC)N1CCC(CSC)CC1 C12(C(C)NC(c3c(CNC(c4c(C)noc4)=O)cc[nH]3)=O)CCC(CO1)C2 C(c1cc(F)c(O)c(F)c1)=CC(N1CCCC(NC(C2(CC=C)CC2)=O)CC1)=O c1(C(N2CCC3(C(CNC(c4cc[nH]n4)=O)C3)CC2)=O)ccc2c(c1)OCCO2 c1(CN2CC(C(=O)Nc3ccc(C(C)O)cc3)C(O)CC2)cc(F)cc(Cl)c1Cl N1(C(CCN(C(C2(C)CC(=O)N(C)C2)=O)CC)=O)CCC2(C1)CC2(F)F O=C(C1CCc2cc(F)ccc21)NCC1CCCN1C(c1n[nH]c2c1COC2)=O CCC(C)CC(=O)NCC1(NC(c2cn(C(C)(C)C)cn2)=O)CC1 c1(C(=O)NC(C)CCN(C)C(C2CCOC2C(F)(F)F)=O)ccc(N)c(O)c1 c1(C(=O)NCCOCCCN(C(c2n(CC)nnc2)=O)C)cc(C)ccc1CC CCC(C)C(=O)C(=O)NC1(C(=O)NCCCF)CCSC1 c1(C(C(=O)NCC(C)CN(C)C(C2(O)CC2)=O)O)cc(F)c(F)cc1F c1(OC)cc(CC(=O)NCC2CCSCC2)ccc1Br.C12CCC(CC1)NC2=O C1(NC(C(Cc2ccccc2)NC(N)=O)=O)CCN(C(C2CC2C2CC2)=O)CC1 CC1CCN2N=C(C(=O)NCC3(F)CC(CNC(C4(Cl)CC4)=O)C3)NC2=N1 c1(NS(CCCC)(=O)=O)ccc(F)c(NC(c2ccc(F)c(C)n2)=O)n1 Cc1ccc(O)c(C(=O)N(C)CC=CC(=O)NCCCc2ncc[nH]2)c1 N1(C(C2CN(C(C)=O)C2)=O)CC2(C1)CN(C(C1CCC(C#N)C1)=O)C2 c1(CNC(COC2(C)CN(C(C3CC(F)C3)=O)C2)=O)ccc(Cl)cc1Cl c1(C(=O)NC2C(NC(=O)OC(C)(C)C)C2)ccc(Br)cc1Sc1cccc(Cl)c1 N1(C(C(C(C)C)C2CCC2)=O)CC2COCC2(C(=O)NCC(C2CC2)C2CC2)C1 C(=O)(CS(=O)(=O)NC)NC(C(=O)NCC(C#C)OC)C1CCCC1 c1(C(=O)NCCCC(C)NC(C(C)NC(=O)OC)=O)c(Br)n[nH]c1C O=C(C1=C(Cl)CCC1)NC(C(N1CC(S(N)(=O)=O)C1)=O)C1CC1 Cc1n[nH]c(C)c1CC(C)C(=O)NCCCCC(C)NC(c1nc(C)n(C)n1)=O C(=O)(C1=NOC(C)C1C)NCC1(O)CCN(C(Cc2cc(C)c(F)cc2)=O)C1 C1(CNC(c2c(C)ncs2)=O)CN(C(c2cnn(CCN(C)C)c2)=O)CC1O c1(OC)ccc(F)cc1CC(=O)NC1CCN(C(=O)C(Br)=C(C)C)CC1O Cc1cc(C(F)Cc2nc(C(C)OC(C)(C)C)nn2-c2ccccc2)ccc1F c1(NC(c2nc(Br)nn2C)(c2nnnn2CCC2(C)CC2)C)ccc(Cl)cc1Cl N1(C(C(CC)OCC)=O)CCC(N(C(=O)CCc2ccsc2)C)C(C)C1 N12CCC(NC3C(CC)C3C)(CC1)COC2=O.C(C)(C)(C)NS(C)(=O)=O c1(OC)cc(C)ccc1N1CCN(c2ccnc(C(F)(F)F)n2)CC1 C(=O)(C1=Cc2ccccc2OC1)NCC1CN(C(C(CCC(C)C)=O)=O)C1 CP(C)(=O)c1ccc(C(=O)NCC2CC2CNC(C2C(C3CC3)C2(F)F)=O)s1 C(=O)(CC1=Cc2ccccc2C1)N(C(C)C)CCNC(C1(C)C=CCC1)=O Cc1cn2cccc(NC(c3csc(NC(=O)Cn4nc(C)cc4C)n3)=O)c2n1 c1(C(=O)NC2CC(NC(CCCC)=O)C2)ccc(Br)c2cccnc12 C1(NC(C(C)CO)=O)CN(C(=O)CN(C)Cc2ccccc2)CC1O N1(C(C(CNC(CCCC(C)=O)=O)O)=O)CCC2(COC(C)C2)C1 c1(CC(=O)NC(C)CCNC(c2cnc(Cl)s2)=O)cn2cccnc2n1 C(=O)(C(O)C(C)CC)N1C(CNC(c2c(C)nc(COC)s2)=O)CC1 C(=O)(C#CC1CCCOC1)NC1CCN(C(C=Cc2ccc(OC)c(Cl)c2)=O)C1 CC1CN(C(=O)CN2CCC(C)C2)CCCN1C(c1ccn2ccnc2c1)=O c1(C(=O)OC)cc(CNC(=O)C(C2CCO2)OC)cs1.C12CC1C(=O)NC2 c1(C(N(CCCCN(C)C(C2(Cl)CC2)=O)C)=O)cc(F)c[nH]1 c1(OCC)cc(CN2CCCC(C)(C(=O)NCCc3cnc[nH]3)C2)ccc1OC c1(C(=O)NC2C(NC(CCSCC)=O)CCC2)cccc([N+](=O)[O-])c1Br C1(NC(c2c(C)oc([N+](=O)[O-])c2)=O)CC2CCC1CN(C(=O)C(C)(C)C(F)F)C2 N1(CC(C(=O)OC)c2ccccc2)CCC(CO)CC(O)C1 C#Cc1cccc(C(=O)NCC2(F)CCN(C(=O)C(CC)n3cccn3)C2)c1 C(=O)(C1CCCc2scnc21)NCCN(C(c1ccc(C(C)=O)o1)=O)C N1(C(C(C)CNC(=O)CCCC(C)C)=O)CCOCC(C)(O)C1 C1(CNC(C2(O)CC(C)(C)C2)=O)(CO)CCN(C(C2CC2C2CCCO2)=O)CC1 c1(NC(C2CCCN2C(C2CCC2)=O)=O)ncc2cc(Br)ccc2n1 C1(NC(=O)C2=CCCCC2)CCCCC12CCN(C(=O)C#CC1CCCC1)C2 c1(NC(C2CC23CCN(C(C2CCOCC2)=O)C3)=O)cnc2[nH]cnc2c1 C(=O)(C#Cc1ccccc1)N1CCC(O)(C(=O)Nc2cccc(C=O)n2)C1 C1(NC(C2CC3(CCC3)C2)=O)CCN(C(c2cnn(C3CCOCC3)c2)=O)CC1 C1(NC(c2ccc(N)c(C)c2C)=O)CN(C(=O)CC2(C)CC2)C2(CCOCC2)C1 N1(C(C(C)SCCCC)=O)CCC(O)(CN(C)C(c2cnc(C)s2)=O)CC1 c1(C(=O)NCC2(OC)CCOC2)ccc2c(c1)C(C)(C)OC2 C(=O)(C(O)CC(F)(F)F)N(CCNC(C1(CCOC)CCC1)=O)C1CC1 Cc1cnc(C(=O)NC2C3CN(C(C4CCN(C5CC5)CC4)=O)CC23)cn1 c1(C(C)=O)cccc(OCCC(N2CC(NC(c3cc(C)c[nH]3)=O)CC2C)=O)c1 N1(C(C(COC)(C)O)=O)CCC2(CCN(C(=O)C(C)C(C)C)C2)C1 C1(CC)C(C(=O)NC2CC(C)(O)C2)CCN1C(c1cc(COC)[nH]n1)=O CC1(C)OC2(C(=O)NCC(C3CC3)NC(c3ccn4cccc4c3)=O)CCC1C2 C(=O)(C1=Cc2cc(C)ccc2OC1)NC1CCC(NC(C2C(C=C)CC2)=O)C1 c1(C(=O)NCC(CNC(c2cc(C)n(C)n2)=O)(C)O)cc(Cl)cc2ccncc12 C#Cc1cn(C)nc1C(N1CCC(NC(C2(NC(C)=O)CCCOC2)=O)C1)=O C1(CNC(CSC)=O)CC2(CC(NC(=O)C(C)Cc3cccc(Br)c3)C2)C1 C#Cc1ccc(C(=O)N(C)CCNC(c2ccc(CC)s2)=O)cc1Cl N1(C(C2CCCN(Cc3cn(Cc4cc(C)no4)nn3)C2)=O)CC(O)CC1(C)C c1(CNC(C(C)C)=O)nnc2n1CCN(C(=O)CC1CC3CC3C1)C2 c1(OC)ccc2c(C(N3CC(NC(c4cccc5occc45)=O)C3)=O)cnn2c1 C(=O)(C1=CCC(C)CC1)N(CC(=O)NCCC(=C)C)CCC C1(O)(C(=O)NCC2CN(C(C=Cc3n(C)ccc3)=O)C2)CCc2ccccc2C1 CN1CC2(CCN(C(=O)C(C)(CNC(C3C=CCS3)=O)N(C)C)CC2)C1 C1(NC(c2c(C(C)C)scn2)=O)CN(C(c2ccsc2)=O)CC2CC12 C12(CNC(C)=O)CC(NC(C3CCCCC34CCC4)=O)(C1)C1(CCOCC1)O2 C(=O)(CCCCC(=O)N1CC2CC(C(N3CCC(CN(C)C)C3)=O)C(C2)C1)OC c1(C(=O)NCC2CCCCN2C(C2CC2(F)F)=O)occ2c1CCCC2 C(=O)(C1=CC2(CCN(C(C3CC3(F)Cl)=O)C2)C1)NC1C(CN(C)C)C1 N#Cc1cncc(CN2CC3CN(C(c4ccc(Cl)nc4F)=O)CC23)c1 c1(C(=O)NCCOC2CCN(C(=O)CC3CC34CC4)C2)cnccc1Br N1(C(=O)Nc2cc(OC(C)C)cc(Br)c2)CC2CCCCC12C c1(CNC(CNC(C2C(C(=O)NCCOC)C2)=O)=O)cccc(Cl)n1 C1(C(=O)NC(c2ccoc2)C)(OC)CN(C(=O)CC2CC(C)=NO2)C1 Cc1cc(O)ccc1CC(=O)N(C1CCCN(C(=O)CCc2nccs2)C1)C C1(C#N)(OC)CC(C(=O)NCCCC(C)NC(=O)CC2CCCOC2)C1 C#CCC(O)C(=O)N1CC(OCC(=O)N(c2cnccc2C)C)C1 c1(CCNC2(C)CC(CO)C2)nc2ccccc2s1 Cc1cc(C(=O)NC2CC(NC(=O)C(C)c3ccsc3)C2)cc(N)c1 c1(CCCNC(C2CN(C(=O)Cc3ccccc3)CCN2)=O)ccc(F)cc1 N1(C(CCOCC)=O)CC(NC(c2ccc3ncncc3c2)=O)CC12CCOC2 c1(C(N(C(C(=O)NCc2cc(C(C)C)no2)C2CC2)C)=O)ccnc(O)c1 CCC(CC(=O)N1CCCC1CNC(c1cc(N)cc(C)c1F)=O)CC(F)(F)F c1(COC)ccc(C(c2nnnn2C2CCC2)Nc2ccsn2)cc1.C1(C)CCCC1 c1(C(=O)OC)cccnc1N1CCOC(COC(=O)COCC2=CC=CN=C(C)S2)C1 N1(C(=O)C(F)n2ccnc2)CC2CC(C(=O)NCCC3CC(F)(F)C3)(C2)C1 CC(CC(=O)NC(CC1CC1)C(N1CCCC(C)CC1)=O)C(F)(F)F Cc1ccc(=N)[nH]c1C(N1CCC(C)(NC(c2ccc(-c3ccco3)[nH]2)=O)C1)=O n1(CC)cc(C(N2CCCC2CCC(=O)NC(C)CN2CCCC2)=O)c(C)n1 c1(NC(C2C(C)CCC2)=O)nc2c(s1)CC(NC(C13CCC(CC1)CC3)=O)CC2 c1(C(c2ccccc2)OC)c[nH]c2ccc(NC(C34CCCC3C4(F)F)=O)cc12 N1(C(C(C)OC(C)=O)=O)CCCC(C)(C(=O)NC(c2nc(C)no2)(C)C)C1 N1(C(C(Cc2ccccc2)OC)=O)CC2C(CNC(c3cnns3)=O)C2C1 c1(N2CCN(C(c3cc(CCC)on3)=O)CC2)nccn(C)c1=O n1(CC)nc(C(=O)N(CCCCC(=O)NCCCCCOC)C)c(C)n1 c1(C(N2CCN(CC)C(C)C2)C(=O)NC2CCC2)ccc2c(c1)COC2 Cc1nc2ccccc2nc1C(=O)NC1C2CCN(C(=O)Cn3nccc3C)C12 N1(c2ccc(C(N(c3cc(I)ccn3)C)=O)cn2)CCc2ccccc21 CC(C)(O)C(F)(F)C(=O)NC1CC(O)CN(C(c2ccc(Cl)cc2)=O)C1 C12(C(=O)NCc3cc(OC)no3)CC(C)(CN1C(c1ncc(F)cn1)=O)C2 N1(C(CN(S(C)(=O)=O)C)=O)CCC(n2cc(CCCCCSC(F)F)nn2)CC1 CC#CCC(C(=O)NC(c1nccn1C)CC)NC(=O)CC(=O)OC c1(SCC(=O)NCC(CC)Oc2ccccc2F)ccc(-c2nn[nH]n2)cc1 C12(C(=O)NC3C(NC(CN(C)C)=O)C3)CCCCC(F)(C1)C2 C1(C(=O)NC(C)CCNC(c2cncn2C)=O)CCCC(C)C1 c1(C(N2C(C(N3CCN(CCCC)CC3)=O)C=CC2)=O)ncnc(C)c1C C1(C)(CNC(c2onc(CC)n2)=O)CCN(C(=O)C=CC2CCC2)C1 Cc1cncc(C(N2CCN(C(=O)Cc3ccn(C)n3)CC2CO)=O)c1C C=Cn1nccc1C(N1C(C(=O)Nc2cn(CCF)nc2C)CCC1C1CC1)=O Cc1cc(O)ccc1C(=O)NC(C)CCNC(=O)C=Cc1cccs1 CN1C(=O)CCC1C(=O)NCC1CC(C)N(C(c2ccc(F)s2)=O)C1 n1(CC)ncc(C(=O)NCC(C)(CO)NC(C2CCC(C(=O)OC)C2)=O)c1Cl C1(NC(CNC(=O)C(C2COC(=O)C2)C2CCCCC2)=O)CC2(CCC2)C1 CCCC(C)(O)CC(=O)N1CCCCC1CNC(=O)C(n1cc(Cl)cn1)C n1(CC(=O)NCC2(F)CCN(C(C(C)N(C)C)=O)C2)ccc2ccccc2c1=O C1(C(=O)NC2C(C(=O)NC(CC)CO)COCC2)CCC(O)CN1C c1(NC(N2CCC(OC(N(C)C)=O)C2)=O)cc(S(=O)(=O)N2CCC2)c[nH]1 c1(C(=O)NCC2CCCN2C(=O)Cc2cn[nH]c2)cccc(C2CC(F)(F)C2)c1 N1(C(C(C)(C)Cl)=O)CCC(C2OCCC2NC(=O)CSCC(N)=O)CC1 N1(C(CSCC(=O)OC)=O)CCOC(C(=O)NCc2oc(C)nc2C)C1 CC1CCN(C(=O)CCc2ccccc2F)C1C(=O)NCCc1nnc(O)o1 CCC(C)(C)C(O)C(=O)N1CC(CNC(c2nccn2C)=O)C2(CCC2)C1 C(CC(=O)NCCC1(O)CCCC1)(C(C)(C)C)NC(CCCNC(C)=O)=O c1(C(C(=O)N(CCNC(=O)CC2CCOC2=O)CC)(C)C)ccc(C(F)F)cc1 C(CC(C)CCNC(c1csc(C(C)C)n1)=O)NC(C1(CC)CCC1)=O c1(CN(C(CC2C(CNC(C(C)NC(=O)OC)=O)C2)=O)C)ccncn1 c1(NC(=O)NCC(CC)OC)ccc(OC)c(C(C)=O)c1 c1(CC(=O)NCCC(C)NC(=O)C(C)n2ccnn2)cc(O)nnc1O C1(NC(CSC(C)C)=O)CCCCCC1NC(c1cnn(C2COC2)c1)=O c1(OC)cncc(C(=O)NCC2(C)CCC(NC(=O)C(C)(C)C3=CC3)C2)c1C C1(CC=C)(C(=O)NCCOCCNC(=O)C(=O)Nc2ccccc2)CCOCC1 c1(NC(C)CS(N)(=O)=O)ccc(S(=O)(=O)NC(Cc2ccsc2)CO)cc1Br C(=O)(CCC(CF)CF)NCc1c(C(=O)NC(c2n(CC)ncn2)C)occ1 N1(C(CC=CC)=O)CCC2CCC(C1)N2C(=O)C(c1cccnc1)OC C12(C(=O)NCC(C(C)(C)O)(C)C)CCCC1CCN2C(=O)CCC1CC1(C)C c1(OC)ccc2[nH]c(=NCCSC)nc(N3CCC(F)(F)C(C#N)C3)c2c1 C12(NC(c3cc(CF)on3)=O)CCOCC1CN(C(C1CCCC(F)(F)C1)=O)C2 Cc1ccc(CNCC(C)N(C)C(c2cccs2)=O)c(O)c1.C12(CC1)C(=O)N2 Cc1c(Br)ccc2[nH]c(C(=O)NCCOCCNC(=O)C=C(C)C3CC3)cc12 Cc1nn(C)c(C)c1NC(=O)Cc1nc(-c2cn(C(C)C)nn2)cs1 C1(OC(C)C(=O)N(C(C)CN(C)C(c2cc(C(N)=O)c[nH]2)=O)C)CCCCC1 Cc1cccc(C=CC(N2CC3(C2)CN(C(c2ccc(Cl)nc2N)=O)C3)=O)c1 c1(C(n2nc(-c3ccccn3)nc2CC2CCCO2)C)c(Cl)cccc1Cl Cc1cccc(C(=O)NC2CC(O)C2CC(=O)N(C)CCn2cccn2)n1 c1(CC(N2CCC(NC(CN(CC#C)C(C)=O)=O)C2)=O)cccc(OCC)c1 C1(O)(C(C)NC(=O)Cn2cc(C3CC3)cn2)CCN(C(C2C(C)(C)C2(C)C)=O)CC1 CP(C)(=O)CN1CC(C(=O)NC2CCN(C(c3c[nH]c(=O)cn3)=O)CC2O)C1 c1(N(CCNC2(CC)CCC2)Cc2ccc(C)s2)nncn1CCOC.CCl C=CCC(C)(C)C(=O)N1CCC(C(C)(C)NC(c2csc(-c3ccoc3)n2)=O)C1 C=C(C)CC(C(=O)N1CCCOC(C)C1)NC(=O)C(N=[N+]=[N-])C(C)C C1(C(=O)NC2C(CNC(c3ccc(C(N)=O)s3)=O)COC2)CC2C(C1)C2(F)F c1(CNC(C(C)C2CCC2)=O)cn(C2CCN(C(=O)C(C)(F)F)C2)nn1 C1(C(=O)NC(c2nc(CC)[nH]n2)C)CC2CC1CN(C(C1(Cl)CC1)=O)C2 C1(C(N(C2CC(C(=O)NC)C2)C)=O)CCC(CCNC(=O)COC(C)=O)O1 C1(CNC(CC(C)CF)=O)CN(C(c2c(C#N)cnn2C)=O)CC12CCOCC2 CCCCC(=O)C(=O)N1CCN(C(c2nc(Cl)sc2Cl)=O)CC1CF c1(OC)ccc(F)c(C(=O)NCCC2(NC(C3CCCC(C#N)C3)=O)CCC2)n1 C12C3CC4C(C3)C14C(=O)N1CC(F)CC1NC(=O)C(C)O2.C1(N(C)C)CC1 n1(CC(=O)NC2C(CNC(c3nc(C(=O)OCC)sc3)=O)C2)ncc(C#N)c1N N1(C(c2cc(C)c(F)cn2)=O)CCCN(C(C2CCCOC2C)=O)C(CO)C1 C#CC1(C(N2CCOCC2)=O)CCN(C(=O)CC=CCN2CCC2)C1 S(=O)(=O)(c1ccc(NCC2CCCC(C)(C)O2)c2cnccc12)NCCCC(C)C C(=O)(CC(C)CN(C)C)NCC(CNC(CC1CC(OCC)C1)=O)CO N1(C(c2cnc(=N)[nH]c2)=O)CCC2(CC1)OCCC2NC(c1cnc[nH]1)=O C1(C(=O)NCCC2CCN(C(C3(C(F)F)CC(=C)C3)=O)C2)CCCS(=O)(=O)C1 C1(CNC(C(C)OCCCC)=O)CCN(C(C2CCC(C)(CC)O2)=O)C12CC2 c1(C(=O)NCC#CCNC(CNC(=O)NC)=O)[nH]c(-c2cccc(C)c2)nc1C C1(C(=O)NC(C)CN(C)C(C2(F)CCS(=O)(=O)C2)=O)Cc2ccccc2CO1 CC(C)(O)C(F)C(=O)NCCC1(O)CN(C(C2CCCOC2)=O)C1 N1(C(C23C(C)OC(CO)(C2)C3)=O)CCCC(F)(CC2CC2)CC1.N12CCCC1C2 C1(CCC)CN(C(c2ccc(N)c(F)n2)=O)CCN1C(C1CCCS1(=O)=O)=O CC(C)C(C)C(C)CC(=O)N1CCCCC(NC(=O)C(C)CCN(C)C)C1 n1(CCOC)nc(C(=O)NCCCN(C)C(c2nsnc2O)=O)ccc1=O c1(NC(C2C(COC)C2)=O)cc2ccccc2nc1C N1(C(CC(C)(C)SC)=O)C(C)CC2CN(C(C34CCC(CC3)C4(C)C)=O)CC12 N1(c2n[nH]c(=NCc3n(C)cc(Cl)c3)s2)CCOc2cccc(Cl)c2C1 c1(C(N2C(CN(C(=O)CC3CCCO3)C)COCC2)=O)ccnc2c1ccn2C C1(C)(C(=O)NC(CC2CN(C(CNC(=O)OC)=O)C2)C)CCCCC1C CCC(C)CC(=O)N1CCC(O)(CN(C)C(c2cncnc2CC(C)C)=O)C1 N1(C(C(C)n2cncn2)=O)CC2(NC(=O)CCCc3ccccc3)CCC1C2 Cc1ccc(C)c(C(N2CC(C)CC2C(N2CCC(=O)C(C)C2)=O)=O)c1O Cc1cccc(C(O)C(N2CCOC(CNC(=O)C=Cc3cncn3C)C2)=O)c1 c1(C(c2n(CC=C)nnn2)NC2(CC)COC2)ccc(OCCC(=O)OC)cc1 C1(CC=C)(NC(=O)Cc2cc(C3CC3)no2)CCN(C(=O)CC2CC=CCC2)C1 c1(C(=O)NC2CCC(NC(=O)CCC3CCCCO3)C2)ccc(Br)cc1F C1(F)(CNC(C=CCCC)=O)COCCN(C(=O)CC2CCC(=O)NC2=O)C1 C(=O)(C1c2c[nH]nc2CCC1C)NCC1(CN(C(C2(OC)CCC2)=O)C)CC1 CCCCS(=O)(=O)CC(=O)N1C2CCC1CN(C(C13CCC(CC)(CC1)C3)=O)CC2 N1(C(C2N(C(c3c(OC)csc3)=O)CC(C)C2)=O)CCCC(C)(OC)CC1 Cc1coc(C=CC(=O)NC(C)CCNC(c2nn(C(C)C)nc2Br)=O)n1 C(=O)(C(F)C(=O)N1CC(OCCC(=O)Nc2nnn(CC)c2C)C1)OCC Cc1ncc(CNC(c2cc(-c3cn(-c4cc(Cl)sc4Cl)nn3)cs2)=O)n1C Cc1cc(-c2cn(CC(C)(C)CNC(C34CCCC3CCC4)=O)nn2)c(C)nn1 c1(C(=O)NC2CCCN(C(C3CC4CCC(C3)S4)=O)C2)sc([N+](=O)[O-])cc1Cl c1(C(N(CCNC(c2c(CC)non2)=O)C)=O)cc(OC)nc2ccccc12 N1(C(c2c(C)c(Cl)ccc2)=O)CCCC(OC(=O)CNC(=O)C(F)C2CC2)CC1 N1(C(=O)NC2C3COCC23)CC2CC1CN2C(c1ccncc1O)=O N(C1CCCc2cc(O)ccc21)C(=O)NCc1ncc(C(C)(F)F)s1 c1(C(CCSC)NC(=O)OCCCNC)nnnn1CCC1CC1 C(CCNC(C12CC1CCN2C(=O)CC1(C)CCC1)=O)(C(C)C)OC c1(OC)cncc(NC(c2ncccc2NCc2cnccc2Cl)=O)c1 C1(NC(C2CCc3ncncc3C2)=O)CC2CCC(C1)N2Cc1cn[nH]c1 N1(C(CC2(C)CC2(Cl)Cl)=O)CCC2CCCC(C1)N2C(=O)Cc1csc(=N)[nH]1 n1(C(C(=O)N(CCNC(CC2CC(OC)C2)=O)CCOCCO)C)cc(Cl)cn1 C1(C(=O)NCCNC(C2CN(C(CN3C(C)CCC3)=O)C2)=O)CSCC(=O)N1 c1(C(N)=O)cccc(C(=O)NC2CN(CC3CC3)C2)n1.c1(CN)ncc(C(=O)O)[nH]1 Cc1ccc(C(=O)NCC(CC(C)C)NC(C2CCC(C)(C)C2)=O)c(Br)c1 C1(N(C(=O)CC=CC(C)(C)C)C)CCC(NC(c2cc(C3CC3)cs2)=O)CC1 c1(C(=O)NCC(CC(F)(F)F)NC(CC2(C=C)CC2)=O)ccc(N)c(F)c1F n1(CC)nccc1C=CC(=O)NC(C1CCOC1)CNC(c1ncsc1CC)=O C(=O)(CC(C)C(C)(C)N)NCCNCCCCC(COC)=O c1(N(C)C)cc(C(=O)OCCc2ccc(CO)o2)ccc1Br c1(OC)cc(Cl)ccc1C(N1CC(CNC(=O)CCC2CC2)C2(CC2)C1)=O C(=O)(C(C)CCCC(C)C)N1CCC(CC(N2C(CO)CC(OC)C2)=O)C1 N(C1CC(C)n2ncnc21)C(=O)NCc1nccc(CC)c1 C1(C(=O)Nc2csc(C(N)=O)n2)CC(F)(F)CN1C(=O)COC1CCCOC1 C=CCCC(C(=O)NC1CC2CCC(C1)S2)NC(=O)C(O)CCCC C1(C(=O)NCC2N(C(c3c(C)scn3)=O)CC2)CC(=O)C12CCCC2 CCC(C)(C)C(=O)NCC(CC(C)C)NC(c1cccc(Cn2cccn2)c1)=O CC1(CNC(c2cnc(C(N)=O)s2)=O)CCN(C(C2(c3cccs3)CC2)=O)C1 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CCOC(CCNC(=O)C=Cc2cn[nH]c2)C1 N1(C(CC2C(C)C2)=O)CC2CCC(NC(C3CC(C)(C)CN3C)=O)CC2C1 N1(N2CCCCC2)CCN(CC(F)F)CC1.CC12CC(C(=O)NC(=O)C(N)=O)(C1)C2 N1(C(C2C(C(C)NC(=O)C(=O)C3CCCC3)C2)=O)CCCC1CN(C)C C(=O)(C(C)CC(=O)N1CCN(C(C2CC2c2cccc(F)c2)=O)C(C)C1)OC CCC(CC(F)(F)F)C(=O)N1CCOC(CN(C)C(c2c[nH]cc(Cl)c2=O)=O)C1 CCCCC(F)(F)C(=O)NC(COC)CNC(=O)C(CC)C(F)(F)F N=c1cc[nH]cc1C(N1CCN(CCCNC(C2(c3cc[nH]n3)CC2)=O)CC1)=O c1(C(=O)NC2CN(Cc3c(C)cccn3)CC2F)cc(C)n(C)c1C C1(N(C(c2ccc(SC(C)C)cc2)=O)C)CCN(C(c2cc(Br)n[nH]2)=O)CC1C c1(CC)ccc(OC)c(C(=O)NC2CC(NC(=O)C(C)C(O)CC)C(O)C2)c1 CC(C)(F)CC(=O)NC1CCC(N2CCN(C(=O)CC3(C)CCCC3)CC2)C1 N1(C(CN(CC)CC)=O)CCN(C(c2ccc(C)c(I)c2)=O)CC(CO)C1 c1(CC(=O)C(=O)CCC(F)(F)F)sc(O)nc1C.C(C(CN)CO)NC(CCNC)=O N1(C(c2nc(COCC)sc2)=O)CCN(C(=O)C(O)CC(F)F)C(CC)C1 C(=O)(CC1CCOc2ccccc21)NCC(C)CNC(c1ccc(O)c(Cl)n1)=O C#Cc1cc(NC(=O)C=CCC(C)(C)NC(c2cnc(OC)nc2)=O)ccc1C c1(C(=O)NCCOCC(F)(F)F)c(F)cc(O)cc1F.C12CCC(CC1)NC2 C(=O)(C#CC1(CC)COC1)NC(CC#C)(C)C(=O)NCc1cnc(O)c(F)c1 CCCCC(O)CC(=O)N1CC2CCC(C1)C2NC(=O)C(C)=C1CCCC1 N1(C(C(F)=C(C)C)=O)CC2(CCC2)CC1CNC(=O)CNC(c1ccc(Cl)s1)=O C1(NC(=NCCC)NCCCc2cccc(Cl)c2)CCC2(C1)OCCO2 c1(C(=O)NC(C2CCN(C(c3cccc(F)c3F)=O)C2)C)ccc(Cl)c(F)c1F Cc1ccc(C=CC(N2CC3C(C(=O)NC4CCCN(C(C)C)C4)C3C2)=O)s1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCOC1)N1CCC(NC(N(CC)CC)=O)C1 N1(C(C2C(C)CCCC2)=O)CCOC2(CCN(C(=O)CC(F)(F)C(F)F)CC2)C1 c1(C(=O)NCCC2(NC(C3CCCSC3)=O)CC2)ccc2c(c1F)CCC2 C(C)(CC=C)(C(=O)NC(CC)C(C)(F)F)NC(c1n(CC#C)cnn1)=O c1(C(N2CCC(O)(C(C)NC(CCCC=C)=O)C2)=O)nccn2cnnc12 C1(C(N2C(c3scc(C(=O)NCC)n3)CCC2)=O)CCCC(C)(C)C1 c1(NC2C(NC(C3(C=C)CCCCC3)=O)CC2)nc(OC)c2ccccc2n1 C=CC(O)C(=O)NCCN(C)C(c1c[nH]nc1C(C)(C)C)=O c1(OC)cccc2[nH]c(C(=O)NC3CN(C(c4ncccc4Cl)=O)CC3F)cc12 C1(CNC(C(CC)OC)=O)CCCCCN1C(=O)CCCc1ccc(F)cc1F C1(NC(CCC)=O)CCCC(CC(=O)NC2CC(OCC)C2(C)C)C1 Cc1cc(C(=O)NCC2(C(N)=O)CN(C(=O)CC3CCOC3=O)C2)no1 c1(CNC(c2ccc(OCC)c(OC)c2)=O)ccc2c(c1)CCCN2C N1(C(C2(COC)CCC2)=O)CC2CCC2(CNC(C2(O)CCCCC2)=O)C1 CC1(C)CCc2[nH]nc(C(N3CCC(NC(C4CC(CCF)C4)=O)CC3)=O)c2C1 C1(CN(C)C(c2csnc2Cl)=O)CCCC(NC(=O)COCCCF)C1 c1(C(=O)NC2CCCN(CC(=O)NCC)C2)cc(C)cc(C#N)c1 c1(C(=O)NC(C(=O)NCC(C(C)C)(C)C)CC2CCCC2)cc(C#N)ccc1N c1(-c2c(COC)cccc2)cnc2c(c1C)N(C(=O)CC(F)(F)F)CCO2 CC1(C)C(NC(c2cscn2)=O)CC1C(N1CC(F)(F)C1)=O N1(C(c2c(C)cn(C)c2)=O)CC2(CCN2C(=O)C=CC(=O)NN2CCCC2)C1 C(C(COC)C(=O)N1CCC(CN(C)C(C2(COC)CC(F)(F)C2)=O)C1)OC N1(C(CC2CCN(C(C(CC)NC)=O)C2)=O)CC2CNCC12 c1(C(N2CC(O)(C(C)NC(C(CC)C(C)O)=O)C2)=O)cccc2c1OCC2 N1(C(C(C=C)(F)F)=O)CCc2[nH]nc(CNC(=O)C(O)CCC)c2C1 C(N=c1[nH]c2c(c(=NCC(CO)C3CC3)[nH]1)SCC2)c1c(Br)ccc(C)c1 C1(C(N2CC(NC(=O)CC3OCCCOC3)C(F)C2)=O)CC2CCC(C1)O2 n1(CC(=O)OC(C)(C)C)nccc1C(=O)NC1CC(NC(C2CC2C#N)=O)C1 N1(C(c2ccc(-c3c(F)ccc(OC)c3)cn2)=O)CCC2(C1)CC2(F)F C1(CC)C(NC(c2ccc(COC)cc2)=O)CCN1C(=O)C1=CCCS1 C1(C(=O)NC(C(=O)OC)C(C)C)CN(C(=O)CN2CCCCC2=O)CC1(C)C C1(C(N(C2CCN(C(=O)CC(C)(O)C3CC3)C2)C)=O)CC2(CCC2)CO1 C1(N(C(CCc2c[nH]c(=N)[nH]2)=O)CCO)CCCN(C(=O)CC2CNC(=O)C2)C1 C(=O)(C1=C(Cl)CC1)N1CCC(N(C(C2(O)CC(CF)C2)=O)CC)C1 CC(O)C(C)(C)CNC(C1CCCC1CNC(=O)CCCC1CCCO1)=O c1(-c2c(C)[nH]cc2)nc(CCO)nn1Cc1cccc(F)c1 c1(C(=O)NCC(C)N(C(CNC(c2c(C)occ2)=O)=O)C)ccc([N+](=O)[O-])nc1 c1(CC(N2C(CC(=O)OCC)C(=O)NCC2)=O)ccc2c(cnn2C)c1 C1(NC(COCCC#C)=O)CCCN(C(c2cnn(C)c2C2CC2)=O)CC1F c1(C(N2CCCN(CCNC(C(C(C)C)O)=O)CC2)=O)c[nH]c2cccc(Cl)c12 c1(OC)ccc(C)nc1C(=O)N(C1CN(C(C2CC(OC)C2)=O)CC1(C)C)C c1(-c2cn(CC3N(C(c4[nH]cc(C)c4C)=O)CCCC3)nn2)cc(Cl)cnc1Cl C1(NC(=O)C(O)CCCc2ccccc2)CN(C(=O)CO)C2CCCC12 c1(C(C)C)ccc(C(=O)NC2CCC2NC(c2cn[nH]c2)=O)cc1 c1(C(N2CCCC(NC(CC(C)CF)=O)C2C)=O)ncnc2ccsc12 Cc1cnc(NC(C2CN(Cc3cccc(N(C)C)c3)C2)=O)cc1Br C1(NC(CN(C2CCSC2)C)=O)CN(C(c2csnn2)=O)CC12CCOCC2 c1(NCC2=C(C)CCCC2(C)C)ccc(N=c2cc[nH]cc2)cc1 C(N=c1[nH]c(Cl)nc2c1CCC2)C12OCC(NC(=O)C(F)C(F)(F)F)(C1)C2 n1(CC)c(CNC(C2CN(C(=O)C3=CCSC3)CC2F)=O)nnc1O N1(C(c2ccc(OC)s2)=O)CCCC2(NC(c3cc4occc4s3)=O)CC2C1 CCCCC(CC)C(=O)N1CCCC(CNC(c2sc(COC)nc2C)=O)C1 Cc1nsc(C)c1C(=O)NCCCN(CCCNC(c1ccncc1F)=O)C N1(C(C(C)c2ccco2)=O)C(CC(=O)NC2C(C)C2C)C2CCCC12 Cc1coc(CNC(=O)C(C)NC(=O)C(C2CCCCC2)F)n1 C1(CNC(C=C(CC)CC)=O)CC(C(=O)N2CCC(OC(C)C)C2)=NO1 N(C1COc2cc(F)c(F)cc21)CC.n12nnnc1C(C)(C1CC1)NC1CC2C1 N1(C(c2c(C)nns2)=O)CCN(C(=O)Cc2ccn(C(F)F)n2)C(C)CC1C C(=O)(C1CCc2ccc(Br)cc21)NC1(C)CCN(C(C2CC(C)(C)C2)=O)C1 c1(CC)nn(C)cc1NC(=O)CC(C)NC(=O)CC1(O)CCCOC1 C1(NC(c2cnc(C3CCCO3)s2)=O)CC2CC1CN(C(C1CC1CF)=O)C2 C1(COC)CCN(C(=O)C(Cn2cncn2)NC(=O)Cn2cc(Cl)cn2)CC1 C1(OCCCCN)CCN(C(=O)C(CC2CCCC2)CN)CC1 C1(C(=O)NC2(C)CCN(C(=O)CCCn3ccnn3)C2)CCOCC12CCC2 N1(C(c2nc[nH]n2)=O)CC=CCC1C(N1CC2C=CC2C1)=O C(=O)(CCC(=O)C(C)(C)C)N1CCCCC(NC(C2C(C)(C)COC2)=O)C1 C1(NC(C2(CF)CC2(F)F)=O)CN(C(=O)CNc2ncccn2)C2(CCC2)C1 C1(CNC(C(c2cnn(C)c2)C)=O)CN(C(=O)Cc2cncs2)CC12CC2 C1(C)(C(=O)N)CC(F)(F)C1.N1(C(=O)OC(C)(C)C)CCCC1C(=O)NC1(CO)CCC1 C1CCCC(=O)N1.c1(C2C(C(N3CCC(NC(C)=O)C3)=O)C2)ccc(C)cc1 C=C1COCCN(C(C2(N=[N+]=[N-])CCN(C(=O)C(C)CO)C2)=O)C1 N(C1CCCc2ccoc21)C(c1cccc(CC)c1)CC(=O)OC(C)=O Cc1cc(C(=O)N(C)CCNC(=O)Cc2cncs2)c(Cl)cc1N O=C(CCCn1cc(C(O)C2CC2)nn1)C1CCCCC1.C12CC1C(=O)NC2=O c1(C(=O)NCC(CCOC)NC(C2CC23CC3)=O)cc(C)c(Br)cc1C C#CCC(CC(=O)Nc1cccc(CC)c1C)NC(=O)CCOCC1CC1 c1(C(N2CC3CN(Cc4cscn4)CC3C2)=O)cn2cc(F)ccc2n1 c1(OC)ccc(CN2CCC(CC(N3CCN(C)CC3CO)=O)C2)c(Cl)c1OC Nc1cc(C(N2CCC3C(NC(=O)Cc4cccc(Br)c4F)C23)=O)cc(F)c1 N1(CCC)CC(C(=O)NC(C)C(C)(C)NC(c2cocc2C)=O)CC1=O N1(C(COCc2cc(C)no2)=O)CCC2(CCCN(C(=O)C(C)CF)C2)CC1 c1(C(N2CC(NC(CC3CCC(C)O3)=O)C2)=O)cccc(N)c1Br N1(C(CSCC(=O)OC)=O)CCC2(CC1)CN(C(C1CC13CC3)=O)C2 C(=O)(C1=Cc2ccccc2C1)N1CCC2(C(CNC(COCCC#C)=O)C2)CC1 N1(C(=O)NCc2ccncc2)CCc2cc(Br)ccc2C1C1CC1 n1(C(C2CCC2)C)nc(Cc2ccccc2)nc1-c1cnn(C(F)F)c1.C1CCO1 N1(C(=O)NCC2CC(=C3CC3)C2)CC2CC1CC2Cc1cc(Br)cs1 c1(C(=O)NCC(C2CCOC2)NC(CCOC)=O)nc[nH]c1C(F)(F)F N#Cc1ccc(NC(=O)C(Cc2ccsc2)NC(=O)CCc2cn[nH]c2)cc1Cl c1(C(N2CCN(CCCNC(=O)CCC3CCC3)CC2)=O)ccc(Cl)c(F)c1F C#Cc1ccnc(C(=O)NCC=CCC(N2CCC23CC(CO)C3)=O)c1 CC(C)CC(O)CC(=O)NCC1CC1CNC(c1cc(CCO)on1)=O C1(NC(C(C#N)=CC(C)C)=O)CN(C(=O)CCc2cc(C)n(C)n2)CCC1C C1(C(N(CCCN(C(CCOC)=O)C)C)=O)CCN(CC(F)(F)F)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(O)(CCNC(C2C(C=C)C2)=O)C1 c1(COC)cc(F)c(C(=O)NCC2C=CCN2C(=O)CO)c(F)c1 CCCC(C(=O)NC1CCC(C(N2CCCC2CCCO)=O)CC1)N(C)C N1(C(C=CCC)=O)CCC2(C(=O)Nc3ccccc3Cl)CCCC12 N1(C(C(C)c2ccco2)=O)CC(CNC(c2cc(O)cs2)=O)C(C)C1 c1(C(=O)NCC(Cc2ccccc2)NC(N)=O)ccc2c(O)nc(S)nc2c1 c1(CC(N2CCCC(N(C(c3nc(C#C)sc3)=O)CC)C2)=O)ccc(C)c(C)c1 C(CCC(C(=O)N1CC(C)C(O)C1)NC(=O)COc1ccccc1)OC c1(CCNC(CN(C(=O)COc2ccccc2)C)=O)nnc2n1CCS2 c1(C(=O)NC2CC(NC(=O)CN3CC4CC4C3)CC2O)cc(F)ccc1Cl CCCC(F)C(=O)NCc1cc(C(N2CCCC(NC(C)=O)C2)=O)co1 CCCCCCCCNC(=O)NC12CC(C(=O)NC3(CN(C)C)CC3)(C1)OC2C C12(CNC(c3ccccc3Br)=O)CCC(C1)N(C(=O)C=CC1CCCO1)C2 C1(CC(=O)NCCc2ocnc2CO)CCC(NC(C2CC2F)=O)C1 c1(CC(=O)NCCN(C(=O)C(C)=C2CCCC2)CC)csc(NC(C)=O)n1 CON=CCC(=O)N1CC=CC(C(=O)NC(C)C(F)F)C1 c1(NC(c2ncccc2NC(c2ccoc2Cl)=O)=O)nc(Br)ccc1C(F)(F)F C(CNC(=O)NCCc1cccs1)(C(C)(C)C)OC CC1(C)CCCC1CN=C(NCC(C(F)(F)F)C1CC1)NC1CCCS(=O)(=O)C1 C(=O)(C(O)C(C)C)NC(CCNC(C1(SC)CC(O)C1)=O)C N1(C(C(C)OCC)=O)CCCC(F)(NC(c2ccc(NS(=O)(=O)CC)cc2)=O)C1 C1(NC(C(C(C)C)SCC)=O)CN(C(C2CCn3nccc3C2)=O)CC(C)(C)C1 C(C(F)(F)C(F)(F)F)n1cc(CNC(CC2C(=O)NCCO2)=O)nn1 c1(OC)cncc(C(=O)N(C)CC2COCCN2C(C23CC(F)(C2)C3)=O)n1 C1(C(=O)OC)CCN(C(=O)Nc2cccc(NC(N)=O)c2)CC1[N+](=O)[O-] CCCCC(CC(=O)N(C)CC1CCN(C)CC1)NC(c1cncn1C)=O c1(CONC(C2C(C)CCN2C(c2c[nH]c(=S)cn2)=O)=O)ccc(F)c(F)c1 C1(CNC(C(F)=CCC)=O)CN(C(=O)C(C2(O)CCCC2)F)CC12CC2 c1(C(N2CCN(CC(=O)NC(CC)C(F)(F)F)CC2)=O)cccc2cnccc12 C(=O)(CC1=NN(C)C(=O)C1)NC(CC#CC)C(=O)NCC1(OCC)CC1 CC1(C)CCC(F)(F)CC1NC(c1cccc2c1C(O)CCC2)=O CC(CC(=O)NCC1(NC(c2cc(CN(C)C)c[nH]2)=O)CCC1)C(F)(F)F O=S(=O)(c1c[nH]ccc1=NCC1CC1)N.c1(NCCN2CCSCC2)ccccc1F c1(OC)ccc(F)cc1CN1CCC(CC(=O)Nc2cccc(I)c2C)CC1 c1(-c2scc(C(=O)NCC3CC3NC(c3nc(Cl)cs3)=O)n2)ccccc1Cl C1(CNC(=O)CCCCNC(C2OC3CCC2C3)=O)CC2CCCC2C1 C1(C(=O)NC2CC3CN(C(C(c4n(C)ccc4)=O)=O)CC32)CC2(C1)CC(C)(C)C2 c1(OC)c(F)cc(C(=O)NCC(C)NC(=O)C(F)(F)c2csc(C)c2)c(N)c1F c1(C(=O)NC2CCC(NC(c3cc(OC)ns3)=O)CC2)c(F)cc(F)cc1Cl C1(C(N2CC(O)(COC)C2)=O)CC(NC(=O)CCCC(C)=O)C12CCC2 c1(CCC)cc(C)c(C(=O)NC(CN(C)C)C(=O)NCc2cn(C3CC3)cn2)o1.CC c1(C(=O)NC2CC(CNC(c3nccc(C)n3)=O)OCC2)ccc([N+](=O)[O-])s1 C(=O)(C(O)CC[S+](C)C)N1CCN(C2CCN(C(c3nccc(C)c3)=O)CC2)CC1 c1(C(=O)NC(CN(C(=O)CC2CCC(=O)N2C)CC)C)cc(S(N)(=O)=O)cnc1C c1(SCC(=O)N(C2CCN(C(=O)C(C)(C)C#N)C2)CCC)cccc(C)c1 CC1CCCC(N(C)C(C2(CNC(c3ccc(C(F)F)o3)=O)CCCO2)=O)C1 c1(C(=O)NCCC(C)N(C(=O)CSC(F)F)C)nc2cnccc2s1 N1(C(C(C)NS(CCCC)(=O)=O)=O)CC2CC1CN2C(=O)CS(=O)(=O)N(C)C c1(C(=O)NC(CNC(CC2N(C)CC=CC2)=O)C2CC2)ccc2nnnn2c1 C1(NC(C=C(C)C(C)C)=O)CC12CCN(C(=O)C1=CCCC1C)CC2 CCC(O)C(C)C(=O)NC1CCCC1NC(=O)CCOCc1ccccc1 Cc1cccnc1-c1cn(CCC(N2CCCC2CC(F)(F)F)=O)nn1 c1(CNC(c2n(CCSC)nnn2)c2ccc(C3CC3)o2)ccccc1N(C)C CC1(C(N2CCCC2CNC(C2CCS(=O)(=O)C2)=O)=O)Cc2ccccc2C1 Cc1cccc(C)c1CNC1CCNC1=O C1(CNC(C(CC)=CC)=O)CC12CCN(C(C1CCn3ncnc3C1)=O)CC2 CN1C2CCCC1CN(C(=O)NCC(c1cc(F)c(Cl)cc1Cl)(C)C)CC2 Cc1ccc(C(=O)NCC(C2CCN(C(C3CC(F)C3)=O)CC2)(C)C)nc1O Cc1cc(OCc2csc(Cc3ccccc3Cl)n2)cc(F)c1 c1(C(=O)NCC2(C(=O)NCC(C(C)C)OC)CCCC2)ccn(C)c(=O)c1 C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NCC(N(C(C(C=CC)O)=O)C)C1CC1 N1(C(C(CCOC)NC(=O)CC(O)C2CC2)=O)CCC(N=[N+]=[N-])CC1 C1(NC(C(C)CN2CCOCC2)=O)CC(C)CN(C(c2ccc(C#N)o2)=O)C1 C1(NC(C(C)n2cccn2)=O)C(C)(C)CN(C(c2ccncc2N)=O)CC1(C)C N1(C(C(C)C)=O)CCN(C(c2cc(OC(F)F)ccc2N)=O)C2CC12 c1(C(N(CC(C)OC)CC)=O)cc(CNC(c2c[nH]nc2C(C)C)=O)on1 c1(CNC(=O)C(=O)C2CC2)ccc2nc(-c3cnn(C4CCCC4)c3)sc2c1 Cn1cnc2c1CCC(C(N1CCCC1(C)CNC(=O)CCc1ccoc1)=O)C2 C(=O)(C1=CCC(C)CC1)NCCCCNC(C(CO)NC(C(C)C)=O)=O c1(CC(=O)NC(CNC(Cc2c(C)ccs2)=O)C2CC2)ccc(N(C)C)nc1 C(=O)(C1CCCc2ncccc21)N1CC(N(C)C(C2C=CC=CC=C2)=O)C(O)C1 c1(CC)cc(N)ccc1C(=O)NC(C)CC1CN(C(C2CC3CC2C3)=O)C1 Cc1cccnc1-n1cc(-c2ccc(CCNC(=O)C(C)OC(C)C)cc2)nn1 c1(OC)ccc(C(=O)NC23CC(NC(=O)C(C4CCOCC4)F)(C2)C3)c(OC)n1 N1(C(c2cnc(C(C)C)nc2)=O)CCN(C(C2CNC(=O)C2)=O)C(CF)C1 Cc1ncc(NC(C2CC(F)CN(C(=O)CN3CCC(C)CC3)C2)=O)cc1Cl c1(NC(c2ccc(CC)cc2)=O)ccc(NC(C2CC(C)(CC)C2)=O)cc1C c1(C(=O)NCC=CCNC(C(C)CC(F)(F)F)=O)c[nH]c2cccc([N+](=O)[O-])c12 C(=O)(C1SCCc2ccccc21)N(CCNC(c1nc(C#C)sc1)=O)C1CC1 C(C)(CCC(=O)N1CCOCC1CN(C)C(c1nccnc1N)=O)OCC Cc1ccc2nc(C(N3CCCN(C(C4CC4F)=O)C(C(C)C)C3)=O)cn2c1 C(c1ccccc1C#N)=CC(=O)NCCCCC(C)NC(c1coc(CO)c1)=O C(=O)(C(C)CCCCCCC)N(CCCNC(C1(CC#C)CCOC1)=O)C1CC1 Cc1ccc([N+](=O)[O-])c(C(N2CCC(C)(NC(c3cc(O)cc(O)c3)=O)C2)=O)c1 C1(CNC(C2C(c3cccc(OC)c3)C2)=O)CC2(CC2)CN1C(=O)CC(C)CF Nc1cc(F)c(CC(=O)NC23CC(NC(C4CCS(=O)(=O)N4)=O)(C2)C3)cc1F c1(C2CCN(C(C3(C)CCCO3)=O)C2)ncc(Br)cn1 Cc1ccc(C(=O)NC23CC(C2)N(C(=O)CCn2cccn2)C3)c2c1NCCC2 O=C(C1=NN2CCCN=C2N1)NC1CC(NC(C2CCCC2C2CC2)=O)C1 c1(C(N2CCC(NC(C(C(CC)O)C)=O)C(F)C2)=O)cc(F)cc2c1C(=O)CC2 N1(C(c2ccc(C)c(C)c2)=O)CCN(C(c2onc(C)c2C)=O)C2CCCCC12 Cc1c(C(=O)NC2(CNC(=O)CC(C)O)CCOCC2)oc2ccccc2c1=O CC1CN(C(=O)CCN(C)C)CCC1NC(C1CCOC1C(F)(F)F)=O CCC(CN(C)C)CC(=O)N1CCCCC1CNC(C1CC1(F)F)=O c1(C(=O)NCC(F)CO)nsc2cc(-c3cnn(CCO)c3)ccc12 N1(Cc2cc(C)nn2-c2cccc(C(F)(F)F)c2)CCC(C)(N2CCCC2)CC1 C1(NC(c2cc(C(C)=O)cn2C)=O)CN(C(=O)C=CC2CC2)C2(CCCCC2)C1 CCCC(CC(=O)NCCC1CC(C)C1)NC(=O)C(F)C1CCC1 C1(NC(CC)=O)CC2CC1N(C(=O)Cc1c(C(F)F)nn(C)c1Cl)C2 C1(CNC(c2c(C)nccc2)=O)CN(C(=O)C(C)(C)C(N)=O)CCC1(C)C c1(OCC(C)C)cccc(C(=O)NC(C)(C)CCNC(C2(C)CC=CCC2)=O)c1 C1(CC)CC(C(=O)NCC=CCNC(C2CCCC2C(N)=O)=O)CC(=O)N1 Cc1cc(C(N2CC(O)(C(F)C(=O)NCC3CCCC(O)C3)C2)=O)cc(C)n1 CC(CC(F)(F)F)N=c1[nH]c(=NCCn2cccnc2=O)[nH]c2ccc(Cl)cc12 C1(C(N2CC3CN(C(=O)C=C(Cl)Cl)CC3C2)=O)CC12CCCc1ccccc12 C12(NC(c3c(C)c(Cl)cnc3)=O)CC3CCC(C1C2)N3C(C1(C)CC=CCC1)=O CC1(C(=O)NCc2ncccc2O)CCCN(C(c2ccc(F)cc2F)=O)C1 CCC(CC(C)C)C(=O)N1CCN(C(=O)CSC(C)C)CC1CS(C)(=O)=O C1(CCC(=O)NC(c2ncc(C)o2)C)CCCCN1C(C1CCC(=O)N1C)=O N1(C(c2ccc(C#C)o2)=O)CCC(C2CCCN(C(=O)C(O)CCC(C)C)C2)C1 O=[N+]([O-])C1CCOCC12CC(F)(F)CN(c1ncncc1F)C2 N1(CC(n2cc(C(c3cnn(C)c3)C)nn2)C)CCC(O)(CO)C1 c1(C(=O)OCC)cnn2ccc(N(C3(CO)CNC3)Cc3ccc(Br)nc3)nc12 Cc1cc2[nH]c(C(=O)NC3CC(C)N(C(c4cn5ncccc5n4)=O)C3)cc2o1 C=CC1CCC1C(=O)NCC1(C(N)=O)CN(C(=O)CCF)C1 C=C1C(OC(c2cc(Br)cc([N+](=O)[O-])c2)=O)CC2CC1C2(C)C CC(C)(C)CC(=O)NCC(N1CCN(CCNC(c2cscc2Cl)=O)CC1)=O C(=O)(CC(CC)CC)N1CC(C#C)(C(N2CCC2C2CCCCC2)=O)C1 C1(C(C)(C)NC(C(C)OCCCC)=O)CCCN1C(c1ccoc1)=O N1(C(C(C(C)(F)F)(C)C)=O)CCC2(C1)CN(C(c1cc(C(F)F)cs1)=O)CCO2 N(C)(S(=O)(=O)N1CC2CCC1CC2)CC#C C1(C(CN(C(=O)C(C(C)NC(=O)CS(C)(=O)=O)C2CCC2)C)O)CC(F)(F)C1 C1(C(N2CC(C)C(n3cc(C4(C)CCCO4)nn3)C2)=O)Cc2nccn2C1 CC1=NOC2(C1)CC(C(N1CCCC(CNC(C3CCCCC3(F)F)=O)C1)=O)C2 CCCS(=O)(=O)C(C)C(=O)NC1CC1CNC(c1cc(N(C)C(C)C)ccn1)=O C(=O)(CC(C(C)(C)C)NC(c1ccccc1)=O)N(C(CC1CC1)CO)C C(C(=O)NN=c1cc[nH]cc1Cl)(C1CCOCC1)N(C)C(=O)OC(C)(C)C C1(CC)C=CCN1C(=O)C(O)C1CN(C(C2CC3CC3C2)=O)C1 CN1CC(O)CCC1C(=O)NC(CC(=O)NCCCCc1ncc[nH]1)C1CC1 c1(C(=O)NCC2C(C)CCN2C(=O)CC2CC(=O)NC2=O)ccn2nccc2n1 c1(C(N2CCC(C)C(CNC(=O)Cc3ccco3)C2)=O)ccn2ncccc12 N1(C(c2c(CC)n(CC)nc2)=O)CCC(CNC(=O)CC2(C)CC2)C(F)(F)CC1 C1(C(=O)NC2(CCNC(C(c3scc(C)n3)C)=O)CC2)CN2CCN1C(C)C2 N1(C(c2c(CC)nns2)=O)CCOCC1C(=O)NCC(C)CN(C)C C1(O)(CNC(=O)CCOc2ccccc2)CCCN(C(=O)C(O)C(F)F)CC1 Cc1cc(C(=O)NCCCC2CCN(C(=O)CC3CC=CC3)CC2)nn1C(F)F c1(C(N2CCC(F)(CNC(C3(Cl)CC3(F)F)=O)C2)=O)cncc(-n2cnnn2)c1 CC(C)(C)C(C(F)F)NC(=O)CC(O)CNC(C1CC2(CCO1)CC2)=O O=C1CC2CC(C(N3CCC(C(F)C(=O)NC4CC4c4ccsc4)C3)=O)C1O2 c1(C(N2C3CC(C(=O)NC(CC#CC)C)(OC3)C2)=O)cnc(C)c(C#N)c1 N1(C(COCC)=O)CCN(C(c2c3c(cc4c2CCC4)CCC3)=O)CC(C)(C)C1 C(=O)(CCCC(=O)N(C)C)N(CC(CC)NC(=O)Cn1nccn1)CC N1(C(C2C(C)(C)CC2)=O)CCC(CCCn2cc(C3CCCOC3)nn2)CC1 Cn1ccc2c(C(N3C(CNC(C4CC(=C5CC5)C4)=O)CC4CC34)=O)ncnc12 c1(C(=O)NC(C2CCN(C(C3(C(C)C)CC3)=O)C2)C)cc(F)c(N)c(F)c1 C(=O)(CC(C)(C)N(C)C)NC(CN(C(c1scc(C)c1Cl)=O)CC)C N1(C(CC=C)=O)CC(CCNC(c2cc(Cl)cn2C)=O)C(C)C1 CC(C)CCC(F)C(=O)N1CCCCC(C(=O)NCC2CC3CCC2O3)C1 c1(CC)ccc(CCC2CCN(C(C3CCC(NCC4CCC4)C3)=O)C2)cc1F N1(C(CCCC#CC)=O)CCC(NC(c2c(C)cc(C)cc2Cl)=O)C(CO)CC1 c1(COC)nc(C)c(C(=O)N(CCCN(C)C(C23CC(C2)C3)=O)C)s1 N1(C(CNS(NC)(=O)=O)=O)CCC(NC(=O)COC2(C)CCC2)C2CC12 C12(C(=O)Nc3cc(C)sc3)CC(CCO1)N(C(C1CC13CCCC3)=O)C2 c1(C(=O)OC)cc(S(=O)(=O)Nc2[nH]c(=N)sc2OC)ccc1I C(=O)(C1=CCOCC1)NCC1CC(C)N(C(c2ncc[nH]2)=O)C1 c1(NC(=O)C(F)CC2CCCCC2)cnccc1Cl.C12(CCCC1)C(=O)NC2 CC(C)C(C)CC(=O)NCC1=CCN(C(C2CCC(=O)N2C)=O)CC1 N1(C(C(CC)=CCCC)=O)CCCC(C(N2CCC(OCCC)C2)=O)(CC)C1 c1(C(N(C)CC2(O)CN(C(C3CC4C=CC3C4)=O)C2)=O)sccc1S(N)(=O)=O c1(C)cc(F)ccc1F.n12nnnc1C(C)(COC(C)(C)C)NCCC2.Cc1nncs1 c1(C(N2C3CC(NC(C(CC)NC)=O)CC2CC3)=O)cc2cc(F)ccc2s1 C(=O)(CC(C)C(C)(C)C)N(C1CCN(C(c2c[nH]c(C)c2)=O)C1)CC c1(C(N(C2CC(C(N3COCC(OCC)C3)=O)C2)C)=O)ccn2ccnc2c1 CN1CC(C)(C)CC1C(=O)Nc1cccc(NC(c2cccc(C(N)=O)c2)=O)c1 C1(CNC(=O)COC(F)(F)F)CC2(CCN(C(=O)CC3=CCCC3)CC2)CO1 C#CC1(O)CCCN(C(=O)COC2(C)CN(C(=O)C(C)(F)F)C2)C1 C(C(C)(C(=O)NC1CCC1CC(=O)NCC1CC(C#N)C1)OC)OC c1(C(N2C(C)(CNC(c3cccc(CC)n3)=O)CCC2)=O)c(Br)cncc1Br C(C)(CNC(=O)C(c1cnn(C)c1)OC)(CC(C)C)NC(C(CC=CCC)C)=O C1(C(=O)NC(C)CNC(=O)Cc2cnoc2)CC12CCOc1ccccc12 C#CCCCCC(c1nnnn1CCCSC)NCCc1scnc1C N1(C(c2cn(CC(C)O)c(=O)cc2)=O)CCC2CN(C(=O)C3=C(Cl)CC3)C2C1 CC1OCCC1C(=O)NCC1CC(C(=O)NCCCC2CCCCC2)C1 CCCCS(=O)(=O)N1CCC(C(=O)NCCNC(=O)CCCOC(C)=O)CC1 c1(C(=O)NC2CCC(NC(C3CC3C(F)(F)F)=O)C2)cnc(C(F)F)nc1 Cc1c(C(=O)NCCn2cc(C(N3CCC(O)(C(F)F)C3)=O)nn2)c[nH]c1C#N N1(C(C(CC(C)C)(C)C)=O)CC2CCC1C1CN(C(=O)CC3=CCCCC3)CC21 C1(C(N2CC(CCC)C(CO)C2)=O)CN(C(=O)CC2CCCOC2)CCN1C C(CCN(C)C(C1CC1F)=O)(C(C)C)NC(CNS(NC)(=O)=O)=O c1(C(C)NCc2cn(C3CC3)nc2C(=O)O)ccc(S(=O)(=O)NC)cc1 n1(CC(=O)NCCCN(C(C(C(CC)O)C)=O)C)c(C(C)C)nc2ccccc12 Cc1cc(C(=O)NCC2CCC2NC(=O)CC(c2c(C)n[nH]c2C)C)sc1C c1(C(N2CCCC(NC(=O)CCCc3nccs3)C2)=O)cc(C(F)F)ccc1F n1(CC)cc(Cl)cc1C(=O)N(CC(CO)(CO)NC(=O)Cc1cnc[nH]1)C CC1(C)C(CNC(=O)CCCc2cnn[nH]2)CCN1c1nccnc1F N1(C(CCC=C)=O)CCCCCC1C(=O)NCCC1CC1C c1(C(N(C)CCN2CCN(C(=O)CCOC3CC3)CC2)=O)ccn2nccc2n1 CC1(C)Cc2cc(C(=O)NCC3C4CN(C(=O)CC5CCOC5)CC34)ccc2O1 c1(C(N2CC(C)C(NC(=O)CC3CC3C)C2)=O)ccnc(F)c1F c1(CN2CCN(C(c3cc(Cl)ncn3)=O)C3C2C3)n[nH]c2c1CCCCC2 CCCCC(CNC(=O)C(C(C)C)N1CCC(C)CC1)NC(=O)COCC(=O)OC CC(C)CC(C)(O)C(=O)N1CCCC(NC(=O)C=Cc2cncnc2O)CC1 C(=O)(C1CCCc2c[nH]nc21)N1CC(C(C)NC(c2c(CC)cncc2)=O)C1 C(N=C(NC1CCN(c2ccc(O)cc2)CC1)NC1CCS(=O)(=O)C1)C1C(=C)C1 N1(CC(=O)NC(c2n(CC)ccn2)C)C(=O)NC2(CCC(C)CC2)C1=O c1(OC)ncc(C(=O)NC(c2ccccc2)Cc2nc[nH]n2)c(C)n1 N1(C(C2CCC(OC)C2)=O)CC=C(CCNC(c2csc(Cl)c2)=O)CC1 CC1CCN(C(=O)C2=NNC(=O)C2)C(CNC(C2COC(=O)O2)=O)C1 c1(C(=O)NCCC(CNC(c2ccc(OC)c(F)c2)=O)O)c(C)cc(=O)oc1C S(=O)(=O)(CCC(=O)N1CCC(C)(NC(C2CCN(c3nccs3)CC2)=O)C1)NC N1(C(COC(CC)(C)C)=O)CCCC2C1CCCCN2C(C1CC(C)(C)O1)=O C1(C(=O)NCC2C3CN(C(c4c[nH]c(=NC)s4)=O)CC32)CC(C)(C)SC(C)(C)C1 N1(C(c2cn(C(C)C)nc2)=O)CC2COCC2(C(=O)NOC2CCOC2)C1 C1(CN(C(=O)Cc2ccc(F)cn2)C)CN(C(C2CC(N3CC(O)C3)C2)=O)CC1O N1(Cc2cn(C)nn2)CC2(CCN2C(=O)CCc2ccccc2)C1 C(C(C(F)(F)F)C(F)(F)F)N1CCN(C2CCCN(C)C2=O)CC1 C1(NC(CCCNC(=O)OC)=O)C2CCC(C2)C1C(=O)NC1CCCC(F)(F)C1 C1(C(N2CC(OCCNC(c3nn[nH]c3Cl)=O)C2)=O)C2CCC1CC2 N1(C(C=C(CCC)C)=O)CCCCCCC1C(=O)NC1CCCCC1(C)C Cc1ncnc2c1OC(C(=O)NC1CC(NC(=O)COCP(C)(C)=O)C1)C2 N1(C(CN(CCOC)C)=O)CCN(C)CC1C(=O)NCCn1cccn1 C1(CN(C(=O)C=Cc2cccnc2)C)CCCCN1C(c1cnc(C2CC2)[nH]1)=O c1(CN(C(c2sccc2C)C(=O)NC(CC)C)C(C)C(C)C)cccc(O)c1 N1(C(CCN(C(C)=O)C)=O)CCN(C)CC1C1CCOCC1 C(CCN=C(NCc1cc(Cl)cn1C)N(C)CC1(c2cccc(Br)c2)CC1)OC N1(C(c2cnc(OCC)s2)=O)CCCCCC(NC(=O)CC2CCOC2(C)C)C1 c1(OC)ccc(C(=O)NC(C2CCN(Cc3cccs3)CC2)C)nn1 CCCCCC(CC)C(=O)N1CC(C(N2CCc3nocc3C2)=O)CC(C)C1 C1(C(=O)NC2(CNC3CC(NC(C4C(C)CN(C)C4)=O)C3)CC2)CC(C)(C)CN1C O=C1NCc2c(C(=O)NC3CC4(CNC(=O)C4)C3)cccc21 C(CC(C(=O)N1CC(CN(C(=O)C=C2CCC(C)C2)C)C1)NC(=O)NC)SC CCCCC(CC)NC(=O)CN(C(=O)C(CC)OC)CCC C1(C(=O)NCC(CCC)OC)CC(O)CN1C(=O)CCc1nncs1 c1(OC)cnc(C(=O)NCC2(O)CC(NC(C3CCC3C(N)=O)=O)C2)cn1 N1(C(C(CC)C(C)C)=O)CC(C)(C)OC2(C1)CN(C(=O)CC1(O)CCCOC1)C2 N1(C(C(C(C)C)NC(C)=O)=O)CCC2(CC1)CN(C(=O)C=C1CCCC1)CCO2 C1(N(C(c2n(C(C)C)nnc2)=O)C)CCCN(C(C2C(C#N)C2(C)C)=O)C1 c1(NCC2(S(C)=O)CC2)nc2ccccc2[nH]c1=NC1CCC2(CC2)C1 c1(C(=O)NCC2CCCCN2C(C2CCCC(F)C2)=O)cc(C2CC2)nc(O)c1 Cc1c(I)c(C(=O)OC(c2ccccc2F)C(F)(F)F)nn1C Cc1nc2c(C)cc(C(N3CCC(NC(=O)C(O)CN(C)C)CC3)=O)cn2n1 CCC(CC)CCC(=O)N1CC(NC(=O)CCC2(C)CC2)CC1(C)C C=CCC(C(=O)NCC(F)CNC(c1nccc(C)n1)=O)NC(C)=O CCC(C)C(C(=O)NCC1CCCO1)N(C1CCCCCC1)Cc1ccccc1 Cc1cccc(C)c1C(O)C(=O)NC1CCC(NC(C2(CC(C)C)COC2)=O)C1 N1(c2nnc(N3CCC(COCC)C3)s2)CCC(C(C)(C)C)CC1 N1(C(c2c(CCC)n(C)nn2)=O)CCCN(C(=O)CCC=C(C)C)CC1 C#CC1(NC(=O)CC2CN(C(=O)CNC(=O)OC)C(C)(C)C2)CCC(C)(C)C1 c1(C(=O)NCCCNC(CC(C)c2ccncc2)=O)ccccc1SCC(N)=O c1(C(N(C)CC2(O)CCN(C(CCSCC)=O)C2)=O)cc2c(cnn2C)nc1C c1(C(=O)NCCC(C)NC(C=CSC)=O)cccc(Cl)n1 N1(C(C(n2cc(Br)cn2)C)=O)CCCC(n2cc(-c3cnc(Cl)s3)nn2)C1 N1(C(CC=C)=O)C2CCCC1CC(CNC(c1ccc(OC)c(OC)c1)=O)C2 Cc1n[nH]c(C)c1CC(N1CC(F)(C(N2CCCC3CC23)=O)C1)=O N1(C(CCc2c(C)cccn2)=O)CC(CNC(=O)Cc2ccoc2)N2CCC1C2 c1(CC(N2CC3C(NC(c4ccc(COC)o4)=O)(C3)C2)=O)ccc(Br)cc1C C1(c2ccc(=N)[nH]n2)NC(=O)N(CC2CCCCO2)C2=C1C(=O)OC2 c1(C(=O)NC2CC(NCc3cn(C)nn3)C2)cccc(C2=CCOCC2)c1 CS(=O)(=O)c1cc([N+](=O)[O-])ccc1N1CCC(NC(C2COCCO2)=O)C(O)C1 N1(C(CC(C)F)=O)CCCC(C2CCN(C(c3cc(C)cc(N)c3)=O)C2)C1 c1(CC=CCC)ccc(C(=O)NCCCNC(=O)C=C2CCN(C)C2)cc1 C12(CNC(CN(C(C(C)C)=O)C)=O)CC1CN(C(c1ccn(C)n1)=O)C2 C1(NC(CCCCN(C(CC2ON=C(C)C2)=O)C)=O)CC2C(C1)C2(F)F C(=O)(C(CC(C)C)NC(C)=O)N(CC(C)NC(c1cccc(C)c1)=O)CC C(=O)(C(O)CC(C)(C)C)N(CCCNC(C(=O)NCC)=O)Cc1ccc(F)cc1 C(=O)(C(C)(C)C(N)=O)NCC1CN(C(c2noc(C)c2C)=O)C1 C(CNC(C1(O)CCC1)=O)(C(C)C(C)C)NC(CCCn1ncc(C)c1)=O C1(NC(=O)CCCC=O)CCN(C(=O)CCC[N+](=O)[O-])CC1F.C(=O)(CCCF)O CC1CN(C(c2cn(C)nc2Cl)=O)CC1NC(=O)CCN1CCCC1 Cc1cc(C(N2CCC(C(=O)N=c3cc[nH][nH]3)C(CO)C2)=O)c(C)n1C(C)(C)C N1(C(c2c(OC)ccs2)C(=O)NCC(C)C)CCC(O)(CN2CCOCC2)C1 c1(NC(C2CCCCCC2)(C)C)ncnc2cnccc12 C1(CCNC(c2cc(C)sc2C)c2n(CCC)nnn2)CCC(F)(F)CC1 N1(C(CC=CC=C)=O)CCCC(C(=O)N(CCCC)CCO)C1 Cc1c2cc(C(=O)NCC(C(C)(C)C)NC(=O)C(C)(C)C)ccc2nn1C c1(C(N2CC(NC(c3cnc(NC(C)=O)o3)=O)C(F)C2)=O)nn(C)c2c1CCC2 C1(CNC(c2ccc(C(CC)(C)C)cc2)=O)CN(C)CCN1C(=O)C(C)CC C#CC1(C(=O)NCCC(C)CCO)CCN(C(=O)CSC)C1 N1(C(c2nc(COCC)sc2)=O)CC(NC(C2(CC3CC3)CCCO2)=O)CC(C)C1 C12(CNC(N3CCC(C(N)=O)C3)=O)CCC(COC1)O2 N1(C(C(COC)NC(C)=O)=O)CCN(C)CC1COCC.C12CCC1NC2=O S(=O)(=O)(CC(=O)NCC1(F)CC(NC(=O)CC2CCCCO2)C1)NC(C)(C)C N1(CC(=O)N(C(c2ccccc2)C)C)CCCC(C)C1CCO C1(CNC(=O)CCc2cnoc2)COCCN(C(c2cn(CCCF)nn2)=O)C1 C(CO)(C(=O)NCC(C)(C)OCC(=O)N(CCCF)C)N(C)C C(=O)(C(F)(F)C(F)F)N1CC(CCc2cn(C3C(OC(C)=O)CCC3)nn2)C1 c12nc(nc3c1CCCCC3)N1CCOC3(CCOC3C1)CC(CC)CCN2C C(=O)(C1CCCc2ncccc21)N1C(C)CC(CNC(C(C=C)(C)O)=O)C1 N12CC(C(C)C1)CN(C(C1CC3CC3C1)=O)C(C)C2=O.C(C)(C)(C)OC(C)=O CCCC(C(=O)N1CCN(C(=O)C(C)CC(F)(F)F)CC1C(C)C)S(N)(=O)=O C12(CNC(COCC(=O)NC)=O)CC1CN(C(=O)C(c1ccc(C)o1)C)C2 C(=O)(CC(O)C(C)C)NC(CNC(CCn1c(C)cc(C)n1)=O)C c1(CNCC(N2C(C)CCCC2)C)ccc(S(=O)(=O)N2CCCCCC2)cc1Br C(=O)(C(CNC(c1cnc(Cl)n1C)=O)C(C)(C)C)N(CC(C)(C)OC)C c1(C(=O)NCC2(F)CCC(NC(C(COCC)C)=O)C2)c[nH]c2nccc-2c1 C1(C)(C(N(CC)CC)=O)CN(C(c2csc(C)n2)=O)CC1C CCC(C)(C)C(C)CC(=O)N1CCC(CCNC(c2cnn(CCO)c2)=O)C1 C1(C(=O)OC)CC2(CC(NC(=O)CC3(C)CCNC3)CCO2)C1 N1(C(CCOCCC)=O)CCN(C)CC1C(=O)NCc1ncc(C)[nH]1 C1(C(=O)NCCN(C(C2CC=CCC2)=O)CC)CCOC2(CCCC2)C1 CCC(CC)C(C(=O)NC1(C(N2CCC(C)(NC(C)=O)C2)=O)CC1(C)C)OC c1(NCC(C)C(F)F)cc(S(=O)(=O)N(C)CCc2ccc(Br)cc2)ccc1C#N c1(N2CCC(N(C(C(CSC)(C)C)=O)CC)C2)ncnc2cccnc12 N1(N(C)C)CCCC(CNC(=O)C(=O)NCC(c2ccccn2)(F)F)C1 N1(C(C(C(C)C)C)=O)CCC(C2(NC(C3CCC(F)CC3)=O)CC2)CC1 c1(C(C(N2CCC(NC(C(C=CCCC)O)=O)CC2)=O)O)ccc(F)cc1C N1(C(C(c2ccccc2Cl)C)=O)CCCOC(CNC(C2CC23CC3)=O)C1 c1(C(=O)NCC2N(C(c3cc(OC)n[nH]3)=O)CCOC2)cncc2c1CCC2 Cc1cccc(CCC(N2CCN(CCCCl)CC2)=O)c1.N12CCC(C1)CC2=O CC1CCN(C(c2cccn2C)=O)CC1NC(=O)Cc1cc(Cl)n(C)n1 C(CC1CCC1)(CC(=O)N1CCC(CC2CCC2)C1)NC(=O)OC(C)(C)C C(=O)(C(CCF)NC(c1cc(C)c[nH]1)=O)N1C(COC)CCC1 C(C(CNC(=O)C(C)(F)CC)C(F)(F)F)NC(c1n(CC)ccn1)=O C1(CC(=O)OC)CCC(C(=O)NCC(C)N(C(=O)CSC(C)C(C)C)C)CC1 N1(C(COC)=O)CCC(NC(=O)CC2CCC2CO)C(C)C1 CCC(C)(C)CC(=O)N(C1CCCCCC1)CCNC(c1cn(C)nc1SC)=O c1(C(N2CCC(C(C)Nc3nccc(C(F)(F)F)n3)C2)=O)ncc2c(n1)COC2 N1(c2n(CCOC)c(-c3[nH]cnc3C)nn2)CCOC(C)(Cc2ccoc2)C1 C1(N(C)C(C2CCC(=O)O2)=O)C=CCN(C(=O)CCOCC(F)F)C1 c1(C(=O)NCC#CCNC(CC2CC(C)C2)=O)cc(Cl)c(F)c([N+](=O)[O-])c1N c1(C(=O)NCC2N(C(c3ccn(CCC)n3)=O)CC2)c[nH]c2cc(F)c(F)cc12 C(=O)(C(=O)CC(C)C)NCC1C(C(N(C(C)C)Cc2ccc(C)cc2)=O)C1(C)C Cn1cc(Br)c2c(NC3CN(C(C4CC(=O)NC(=O)N4)=O)CC3O)ncnc12 CC1CCN(C(=O)CCN(C(C2CC3(C2)CC(O)C3)=O)CC2CC2)CC1C C12(C(=O)NC)CC(CNC(=O)CN(C)C(=O)OC(C)(C)C)(C1)OC2(C)C c1(C(=O)NCC2(O)CN(Cc3n[nH]c(=N)s3)C2)c(Cl)ccc2c1OCO2 c1(NC(C2N(C(C(c3ccc(Cl)cc3)OC)=O)CC(F)C2)=O)cc(Cl)cc(Br)c1 c1(CC(=O)NCC23CC2CN(C(=O)CC2C=CCC2)C3)ccc(C(F)F)cc1 C1(NC(c2ccc(OC(C)C)nn2)=O)CCC12CCN(C(=O)CC1CC1)CC2 CCC(C)CCCC(=O)N1CC(C)(C)CC1CC(=O)Nc1ccc2c(c1)OCO2 CC(C)C(C(=O)NC(CCO)C(F)(F)F)C(C)NC(c1cccc(F)c1)=O c1(CC(=O)NCC2(O)CN(C(C(C=C)(C)O)=O)C2)ccc(C)c(C)c1 C1(NC(c2ccon2)=O)CN(C(=O)CC2CCCCC2O)CCC1CO C1(NC(C2CCN(OC)CC2)=O)CCC2(CC1)CC(NC(=O)C(C)CF)C2 CC1CN(C(=O)CC2CN(C)C2)CCN1C(=O)CCCOc1ccccc1F C1(NS(C)(=O)=O)(CNC(C2CCCC2)=O)CCOCC1.C1(C(=O)N)CC1F C1(CNC(=O)CC2CC2(Cl)Cl)CC2(CCC2)CN1C(=O)COc1ccccc1Cl c1(CNC(CC)=O)cc(C)c(C(=O)NC(C)(C)CC2CCCC2)o1 Cc1ncc(C)c(N2CCN(C(=O)CCOc3ccccc3)CC2)n1 C1(C(=O)NCC2(O)CN(C(C=CCCC(C)C)=O)C2)CCCC1C1CC1 N1(C(C(CCC)C)=O)CCN(C(c2cscc2F)=O)C(CC(F)(F)F)C1 C1(NC(CCCC=C)=O)CCN(C(=O)Nc2cc(OC)cc(O)c2)CC1C C1(CNC(CCNC(COC)=O)=O)CCC2CN(C(=O)C(F)(F)C(F)F)CC12 Oc1nc2nc(-c3cncc4ccccc34)ncc2o1 N#Cc1c(N2CC(CCCCNC(C3CC34CCC4)=O)C2)ncc2c1CCC2 CCC(C(=O)N(CC(C)N(C)C(C1(COCC)CCC1)=O)C)SC n1(C(C)C)cc(C(=O)NCCN(c2cnc[nH]2)C(c2ccccc2)=O)ccc1=O C1(C(=O)NCC2(COC)CCC2)C(NC(C2CCS2(=O)=O)=O)C1(C)C C1(C(=O)NC2(CC=C)CCC2)CCN(C(c2ccc3cc[nH]c3c2)=O)C(C)(C)C1 c1(C(=O)NCC2(C)CCCN2C(C2CCCC2(F)F)=O)cc(F)cc(F)c1 c1(C(=O)NCCN(C(C2CC2CN(C)C)=O)CC)ccc(S(N)(=O)=O)cc1N N1(C2(CCCCNC(=O)CCc3cnn[nH]3)CC2)CC2C(C1)C2(F)F C1(C(=O)N(c2ccc(Cl)cc2)CC)(O)CC2CCC1CC2.C(=O)(C#CC1CNC1)CC c1(C(=O)NC(C)C(c2ccccc2)NC(=O)Cn2cccn2)c[nH]nc1C(F)F c1(NC(N2CC(C(=O)OC)C(F)(F)CC2)=O)ccc2nccnc2n1 c1(-n2cc(CN(C(C(=C)C)=O)CC(=O)O)nn2)ccc(-c2ccc(F)cc2)cc1 C1(NC(C(N2CC(C)C2)C)=O)C(C(=O)NC2CN(CC(F)F)C2)C1(C)C CC1C(CO)N1C(=O)OC(C)(C)C.C1C(F)CN1 N1(C(=O)Cc2ccc(F)cc2F)CC2CCC(C1)N2CC1CCCS(=O)(=O)C1 NC1CCC(N2CCN(C(=O)C(N3CCC(CN)C3)=O)CC2)CC1 CC1CCN(C(=O)Cn2ncn(C)c2=O)CC1CNC(=O)CSC1CCCCO1 c1(OCCC(N2CC(O)(CNC(c3c(CC)ccs3)=O)C2)=O)ccc(C)cc1C C1(C(=O)NC(c2scc(C)n2)C)CN(C(c2cccnc2)=O)CC1C1CC1 c1(OC)ccc(C(=O)N(CCC(C)NC(c2coc(C)c2)=O)C)c(OC(C)C)c1 C1(NC(C)=O)CCCCN(C(=O)COc2cc(C3CC3)nn2-c2ccccc2)C1 c1(CC)cc(=NC(=O)c2c(C)nc3sccn23)[nH]o1 c1(CNC(=O)COCCNC(=O)CN2CCSCC2)ccc(CO)cc1 C1(NC(C(c2n(C)ncc2)O)=O)CCN(C(=O)Cc2ccno2)CC1 c1(C(N2CC(NC(c3ccc(C)c(Br)c3)=O)C(C#N)C2)=O)cc(Cl)c(O)cc1F Cc1cc(C(=O)NCC2(C)CN(C(=O)CC3CC4(CC4)CO3)CCO2)cc(N)c1 c1(CC)ccc(NC(=O)CSCCNC(C2(Cl)CCC2)=O)cn1 c1(C(N(CCNC(c2c(C#C)cn(C)n2)=O)C)=O)c(F)cccc1[N+](=O)[O-] c1(CC(=O)NCCCC(C)NC(c2cc(F)ccc2Cl)=O)ccc(F)cc1F c1(CN(C(=O)C(=O)NC2CC(C(=O)O)C3CC23)C)nn(C)c2ccccc12 C1(NC(=O)NC(C=CC(=O)OCC)C)CCc2cc(OC)ccc2C1 CN1CCCC(CNC(C2CC(CNC(=O)CN(CC(=O)NC)C)C2)=O)C1 O(CP(C)(C)=O)CC(=O)NCC(C)NC(=O)CSc1nnnn1C1CCCC1 N1(CC(C)(C)NC(C(Br)=C(C)C)=O)CCN(C(=O)CC2CC2C)CC1 CC(CC(=O)NC1CCC2CC1CN2C(C1CCN(C)CC1)=O)CC(C)(C)C N1(C(c2c(C)n(C)cc2)=O)CC2CCC(CNC(C3CCOC3(C)C)=O)(C2)C1 C1(C(=O)NCC=CCNC(=O)Cc2cccnc2)CC2(C1)CS(=O)(=O)C2 C(=O)(C(F)(F)CNC(=O)CCCc1c(C(F)(F)F)coc1C)OCC C1(O)(CN(C(C(C)=CC)=O)CC)CC2CCC(C1)N2C(=O)C(C)Cn1ccc(C)n1 N1(C(CCCCC=CC)=O)CCc2ccccc2C(NC(c2csnn2)=O)C1 CC1CC(C(=O)NC2CCNC2=O)CCN1C(C1CC(O)CN1C)=O N1(C(=O)Cc2cccc(Cl)c2F)CCN(C(c2c(Cl)cncc2Cl)=O)C2CC12 N1(C(=O)CC2CC(C3CC3)C2)CC2CN(S(=O)(=O)C(F)(F)F)CC2C1 C1(O)(CNC(C(COC)C)=O)CCN(C(c2ccc(=O)n(O)c2)=O)CC1 C(=O)(C1=NOC(CNC(=O)CNC(C2CCCC2)=O)C1)NCC(CSC)OC c1(C(=O)OCC)ccccc1C(N(C1CC(CCSC)C1)C)=O CC1(CNC(c2csc(Cl)n2)=O)CN(C(=O)Cc2cccs2)CCO1 C(CN=c1cc(C)[nH]c(=NCCn2ccccc2=O)[nH]1)N(CC(=C)C)C C1(O)(CNC(CCc2c(C)noc2)=O)CCN(C(=O)CCOCCN(C)C)C1 c12c(ccc3c1CCC3)NC2=O.c12cn(nn1)CC1CCCN1C(=O)C2.CO C1(CNC(C(c2ccccn2)C)=O)CC2(CCC2)CN1C(=O)CCOCC(F)F C12(C(=O)NC(C=C)(C)C)CCCC1CCN2C(=O)CCCOC C1(C(F)F)(CNC(C2(C)C=CCC2)=O)CCN(C(=O)COC2CCCC2)C1 CCCCC(F)C(=O)NCC(CCOC)NC(=O)C(C)c1cc[nH]n1 C(=O)(C(F)(F)C(C)(C)O)N1CCCC(C(N2CCNC(=O)CC2)=O)(CC)C1 Cn1cc(C(=O)NC2CCCC(CNC(=O)Cc3ccccc3)C2)c(C(F)F)n1 N1(C(=O)CN(C(=O)C(F)C2CCCC2)C2CC2)C2CCC1CC1(CC1)C2 C1(C)(C(N(C(C)C(=O)NC2CC(CCSC)C2)CCC)=O)CCCC1 C1(C(N2CCC(CN(C(=O)CNC=O)C)C2)=O)CC12CCC1(CC1)CC2 N1(C(c2ccn(CCNC(C(C=C)CC)=O)c2)=O)CCC(CO)=C(F)C1 C1(CNC(CC2(C)OCCO2)=O)CCC(C(=O)NC2CCCN(CCO)C2)CC1 Cc1nc(NCC(c2ccncc2F)(C)C)cc(=NCC(C(C)(C)C)N(C)C)[nH]1 N1(C(C2(OC)CC2)=O)CC2CC(C1)CN(C(c1[nH]c(=N)ccc1Br)=O)C2 Cc1sc2cc(F)ccc2c1CCNC(C1(c2cc[nH]n2)CCOCC1)=O S(=O)(=O)(c1cccc(C(N2CC(c3c(F)cccc3F)(O)C2)=O)c1)N(C)C CN1CC(O)CC1(C)C(N1CC2(C1)CN(C(C1CC1(C)Br)=O)C2)=O c1(CCC)nnc(N(C)Cc2ccnn2C)n1CC1CCCO1 c1(NC)ccc(C(N2CCCCC2C(=O)NC(C)(CO)C(C)(C)O)=O)cc1 C1(C)(CC(=O)NCCC(=O)N(CCC)CCS(=O)(=O)CC)CC(F)(F)C1 CCC(C)C(O)C(=O)NCC(C(C)C)NC(c1ccc(C)c(OCC=CC)c1)=O Cc1c(Br)c(C(=O)N(CCNC(=O)C(c2cnccn2)C)C(C)C)nn1C c1(-c2scc(NC(C3CCCN3CC(F)(F)F)=O)n2)ccc(F)cc1 N1(C(C2C(C)C2C)=O)CCc2c(CNC(C3(F)CCCCC3)=O)cccc2C1 C(c1ccc(F)cc1[N+](=O)[O-])=C(C#N)C(=O)NC1CC(NC(=O)C=CCF)C1 c1(C(C(=O)N(CCOCCCNC(C2(CC)CC2)=O)C)C)c[nH]c2ccccc12 c1(NC(C2(C)CCCN2Cc2cc(O)nc(O)n2)=O)c(Br)cc(F)cc1[N+](=O)[O-] C123COC(C1)C(C2)N3.N1(C(C)=O)CCCCC1CCC(C(=O)C(F)(F)CO)=O CC(C)(C#N)CCC(=O)NC1CCCC1NC(c1scnc1C1CC1)=O N1(C(CNC(=O)NC)=O)CCC2(OC(F)F)CC2C1.c12ccc(c(C)c1)[nH]c2=O C(=O)(CCOC)N(CC(C)NC(C1C(CC)C1)=O)CC Cc1cc(CC(N2CCC(O)(C(C)NC(c3cccc(CO)c3)=O)C2)=O)n(C)n1 c1(CC(=O)NCC(CC=C)NC(C2(C)CCCCC2)=O)ccc2ccoc2c1 c1(C(N(CC(C)O)CCNC(C(C)SCC)=O)=O)ccc(CO)c(F)c1 Cc1cn2c(CC(N3CC4(CCC4NC(C4CC45CCCC5)=O)C3)=O)csc2n1 C1(C(=O)NCC(CSCC)(C)C)CSCCN1C(=O)OC(C)(C)C Cc1cccc2cc(C(=O)NC3CC3CNC(=O)C(C#N)C3CC3)oc12 N1(C(C2C(=C)C2CO)=O)CC2CC2(NC(C2C(C(=O)NC(C)=O)C2(C)C)=O)C1 N1(C(C(CC)(C)C)=O)CC2CS(=O)(=O)CC2(NC(c2ncc(C)cc2OC)=O)C1 C(CC(=O)NC1CCCC(O)C1)(C(F)(F)F)NC(c1cc(C)cc(C)n1)=O c1(C(=O)NCC(C)(C)NC(C(C)NC(=O)NC)=O)ccc(C(N)=O)[nH]1 c1(NCC2N(C)CCN(C)C2)ccc(S(=O)(=O)NC2CCSC2)c(Cl)c1 CC1(CNC(c2cc(Cl)cs2)=O)CCCN(C(=O)C=CC2COC(C)(C)O2)C1 c1(C(=O)NC(C)CN(C(=O)CCNC(N)=O)C)nc[nH]c2nccc1-2 N1(C(c2nnn(C)c2N)=O)CC(C(=O)NC2CN3CCCC2C3)CC1(C)C CCCS(=O)(=O)C(C)C(=O)NC1CCN(C(=O)COCc2cccc(OC)c2)C1 Cc1cc(C(N2CCC(C(C)(C)NC(C3(C4CCCO4)CCC3)=O)C2)=O)c(C)s1 c1(OC)cnnc(C(=O)NC2(CCCC(=O)N(CC(C)O)C(C)C)CCC2)c1 N1(C(C(CC(C)C)ONC(=O)Cn2cc(Cl)cn2)=O)C2CCC1CC1(C2)N=N1 N1(C(c2c(COC)noc2)=O)CCCC2CN(C(c3nncs3)=O)CCC12 c1(OCC)c(CC(=O)N(CC(O)CNC(c2[nH]c(C)nc2C)=O)C)cccc1Cl N1(C(COC(C)=O)=O)CC2C(C1C(=O)Nc1ncccc1C(N)=O)C2(C)C C1(NC(c2nc(COCC)sc2)=O)C2CCC1N(C(=O)C(C)CO)C2 N1(C(C2CC(CC)C2)=O)CCC(C(=O)NC(c2ccccc2F)C)(CO)C1 N1(C(c2c(OC)scc2)=O)CCCCC1CC(=O)NCCN(C)C(C)C c1(C(=O)NCC2C(C)CN(C(C3C=CCC3)=O)C2)nc(Cl)ccc1N C1(CNC(CCNC(C)=O)=O)CCC2CN(C(c3ccn4nccc4c3)=O)CC12 C1(CC(=O)NCCOCCOC)CC(NC(c2nnsc2C(F)F)=O)C1(C)C C1(C(N2CC(C)(C(=O)NCc3n(C)ncc3)C2)=O)CC2(CCC2)C1 N1(C(COC2CN(C(COC(CC)(C)C)=O)C2)=O)CC(C)C12CCOCC2 N1(C(CCNC(NOCCCNC(=O)OCC)=O)=O)CC2(C)CCC2(C)C1 N1(C(C(=O)NC2CCOC2)CC2CC2(Cl)Cl)CCC2(CC1)CC2(F)F c1(CC(C(=O)N(C(C)CCNC(c2cc(Cl)on2)=O)C)O)cccc(Cl)c1 CC1CCC(N(C(c2ccccc2)(C)C)C(=O)Cc2ccccc2Cl)CN1CC#N C1(C#N)(NC(c2c(C)nn[nH]2)=O)CCN(Cc2cccc(I)c2O)C1 c1(C(N2CC(C(C)NC(C3CCSCC3)=O)C2)=O)c[nH]c2nc(Cl)ccc12 c1(NC(N2CCCC2c2ccccc2)=O)cccn2ncnc12 C1(NC(CCCC#C)=O)CC2CC1CC2C(=O)NCC(C)SC N1(C(c2ccc(C(C)C)o2)=O)CC2(C)CC1(C(N(C1CCC1)CCO)=O)C2 c1(CS(C)=O)cccc(C(=O)N(CCNC(C2CCC2F)=O)C2CC2)c1 N1(C(c2[nH]ccc(=N)n2)=O)CC2CN(C(C3(F)CCOC3)=O)CC2C1 CCC1=NOC(CC(N2CC(O)CC2CC(=O)NCC(F)Cl)=O)C1 c1(C(C)C)nc(-c2cccc(OCC(N)=O)c2)cc(=NCC(F)(F)F)[nH]1 CC(CN(C)C)CCC(=O)N1CCC(NC(C2CN(C3COC3)C2)=O)C12CC2 c1(COC(C(=O)NCC(CC)NC(C2(C(N)=O)CCC2)=O)C)ccc(C#N)cc1 c1(NC2C3(CC(OC)C3)C2)nc(NC(C)CC(C)C)c2cnn(C)c2n1 c1(C(=O)OC)c(C)cc(C)nc1NC(C)CN(C(=O)C1=CCCO1)C Cc1cc(N)ccc1C(N1CC(C)(C)CC1CNC(=O)Cc1cccnc1)=O C1(CNC(c2c(C)scn2)=O)CN(C(c2cnc(O)o2)=O)C2CCN1C2 CCCCCCC(=O)NC12CC(C1)N(C(C1CCCNS1(=O)=O)=O)C2 c1(CC#N)ccc(C(=O)NCC(O)CC(=O)NC2CCCSCC2)cc1 c1(C(N2C(CNC(c3c(N)csn3)=O)CC2)=O)ccc2c(c1)OCCCO2 n1(CC(N2C3C(NC(=O)CC4CCCCO4)C(C3)C2)=O)ccc([N+](=O)[O-])n1 N1(C(C2C(C=C)C2)=O)CC2CCN(C(=O)CCOc3ccccc3)CC2C1 N1(C(C2(C)CC(C)C2)=O)CCN(C(=O)C(c2ccn(C)n2)C)C(C(F)F)C1 Cc1cccc2c1c(CCNc1cc(=NCc3nnnn3C)[nH]cn1)cn2C c1(C(C)C(=O)NCC(C)NC(=O)COCCc2ccccc2)cc(F)cc(F)c1 Cc1cc(CNC(C2(NC(=O)C(C3CCOCC3)C)CCCCC2)=O)ccc1O N1(C(CCC#CC)=O)CC(NC(=O)CCN2CCC(C(N)=O)CC2)CC(F)C1 N1(C(C)=O)CCCC(C(=O)N(C(CNC(=O)C=CI)Cc2ccccc2)CC)C1 C(=O)(CCP(C)(C)=O)N1CCC(C)(CNC(CC(C(C)C)c2ccc(Cl)cc2)=O)C1 Cn1cnc2c(N3C4CCC3CC(F)(F)C4)nc(=NC3CCOC3C)[nH]c12 O=C1Cc2ccnc(N3CCN(C(C4(CC(=O)OC(C)(C)C)CC4)O)CC3)c2N1 Cc1nc(C=CC(=O)NC(C)C(C)(C)NC(C2CC(F)(F)C2)=O)cs1 N1C2CCc3cc(C(C(N4Cc5ccccc5C4=O)CC)=O)c1cc32.OC C1(NC(C2(C)CC2)=O)CN(C(=O)CCS(=O)(=O)Cc2ccccc2)CC2(CC2)C1 CCCCCCC(C)C(=O)N(C(C)CC(N1C2CSCC1C2)=O)C CC(C(C)(C)C(=O)NCC1(C)CNC(=O)O1)NC(C1CNC(=O)O1)=O Cc1cc(N2CCC(CCNC(c3cc(=O)cc[nH]3)=O)C2)n2ncnc2n1 C1(OC)CN(C(C2(NC(c3cnc(N(C)C)cn3)=O)CC(F)C2)=O)CC12CC2 C1(C(=O)NCC(=O)N(C)CC)CCCCN1C(c1c[nH]c(=NC)s1)=O C(c1ccc(O)cc1)=CC(N1CCC(c2ccccc2)(NC(C(C)C)=O)C1)=O Cc1nc(O)nc(O)c1NC(C1CC(O)CN1C(c1c(Cl)cc(Br)cc1Cl)=O)=O N1(C(=O)CSCc2ccncc2)CCC2(C1)CN(C(C1CC(F)C(=O)N1)=O)C2 c1(C(N2CC(CC(C)NC(C3(C#C)CCCC3)=O)C2)=O)cccc(=S)n1O C1(C(N(C)CC2OCCN(C)C2)=O)CC(O)CCN1C(C1COCCO1)=O N12CCC(O)C(C1)C(=O)NCC2=O.Cc1cccc(COC(C2(CO)CC2C)=O)c1 C1(C(N(CCCOCCNC(C2CCC(CC)CC2)=O)C)=O)CCC(C)=C(C)C1 CC(C)(CCCCNC(=O)CCCF)NC(C1CS(=O)C1)=O C12(C(N3CC(NC(c4ccc[n+]([O-])c4)=O)C(O)C3)=O)CCCC1C2(F)F CC1(C)C(CO)CN1C(C1COCCC1NC(=O)C=CCN1CCC1)=O C1(CC)CC(C(=O)NCC2CCC(CC)CC2)CCO1 C(C(F)C(=O)N1CCC(CC(F)F)C1)C1CN(C(C2(OC(C)=O)CC2)=O)C1 CCS(=O)(=O)CC(=O)N(CCN(C)C(C1(C(N)=O)CC1)=O)C(C)C C12(C(=O)NC(C(C)C)CCN(C(=O)C(=O)NC3CC3)C)CC(C)(CCO1)C2 c1(CNC(CCC(C)NC(C2C3CCCC23)=O)=O)cccc(O)c1F N1(C(CCC)=O)CCC(NC(c2csc(C(C)=O)n2)=O)C(F)C1 N1(C(CC2CC(CC)C2)=O)C(C(=O)NCC(C)Cn2ccnc2)CCC1C N1(C(CN2C(C)CCC2)=O)CCSCC1C(=O)NC(CC1CC1)C1CC1 N1(C(C(C)OC)=O)CCC2(CCCN2C(=O)Cc2nc(C)sc2Cl)CC1 N1(C(C(C)N(C)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1c1ccccc1 N1(C(c2ccc(CC)s2)C(=O)NCCCN2CCCC2)CC2CC(O)CC1C2 N1(C(C(C)N2CCCC2)=O)CC(C(=O)Nc2ccn(C)n2)CC12CCC2 C1(C(N2CCC(C(=O)NC3(CC(=O)OCC)CC3)CC2)=O)CC(=O)NC(C)C1 c1(C(C(=O)NC2CC(C)(NC(c3c[nH]nc3F)=O)C2)O)ccc(Cl)cc1Cl C(=O)(C(O)CCC[N+](C(C1CS(=O)C1)=O)([O-])N(C)C)N1CCCC(COCC)C1 c1(NC(c2c(-c3c(C)cc(OCC)nc3)csc2)=O)ccc2nc(O)oc2c1 C1(C(F)(F)F)(NC(=O)CCOC(F)(F)F)CN(C(c2csc(C3CC3)n2)=O)C1 C(=O)(C(C)(CC)CO)N(CCCNC(C(CCC)C)=O)C S(=O)(=O)(c1cccc(=NCCCCSC)[nH]1)N(CC(CC)Nc1ccccc1)C c1(C(=O)NC2C(NC(=O)CCNc3nccs3)CC2)cc(Cl)no1 C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)NC(C=C(C)c1cccc(Cl)c1)=O N=c1ccnc(N2CCN(C(c3ccc(N4CCOCC4=O)cc3)=O)CC2)[nH]1 N1(CCC)CCCCC1C(=O)C(C1(CNOC)CC1(C)C)=O.C1(CNC=O)CCC1CO C1(CNC(C(C2CCCCC2)OC)=O)C2CN(C(c3snc(O)c3Cl)=O)CC12 C1(OC)C(NC(=O)CCC2(C)CN(C(=O)COCC3CCC3)C2)CC1(C)C c1(CC)cc(C(=O)NCCCC(C)NC(c2coc(O)n2)=O)cc(C(F)(F)F)c1 C1(NC(c2c(CC)n(CCO)nc2)=O)CN(C(C2(SC)CC2)=O)CCC1C C1(CNC(c2cc(CC)c(C)s2)=O)CN(C(=O)C2=CCCS2)CCC1(C)C c1(C(=O)NC2CCCN(C(C3C(OC)CCC3)=O)C2)cc(F)c(F)c(O)c1F N1(C(CCc2ccc(SC)cc2)=O)CC(=O)NC2CN(C(C3CC3C)=O)CCC12 C1(OCC(=O)N(CC(O)CO)CCO)CCN(C(=O)Cc2nnn(C(C)(C)C)n2)C1 c1(CC)nc(C(=O)NCC(O)C(=O)NCCC(C)CO)cs1 Cc1cc(F)ccc1-c1ccc(CN2CCOC(C)(C)C2)cc1 O=C1CC(C(=O)NCc2cn(C3CCCN(C(=O)C4=CCC4)C3)nn2)CCN1 c1(NC(=O)NC2CC3CC(C(=O)O)CC3C2)noc2c1CCCCC2 C1(C(=O)NCC(C)(C)NC(c2csc(Cl)n2)=O)Cc2ccccc2OC1C(F)F CCC(C)(CCNC(=O)Cc1ccns1)NC(C1CC2(CC2)CO1)=O C1(C(=O)NC(c2cccc(OC)c2)C2CCSCC2)CCC(=O)NC1C c1(NS(CNC(CCCCCC#C)=O)(=O)=O)ccc2c(c1)n(C)c(=O)n2C c1(CC(C)C)ccc(C(N2CCN(C(=O)CS(N)(=O)=O)CC2)=O)cc1 C1(C(=O)NC2(CNC(C(CC)c3ccccc3)=O)CCC2)CCCC(C)(C)CC1 Cc1[nH]nc2c1CCN(C(C)C(=O)NCCc1ccnc(C(N)=O)c1)C2 Cc1cnc(C(N2CC3CC2CN3C(C2COC3(CO)CC2C3)=O)=O)cc1Cl N1(C(c2c(SC)n(C)nc2)=O)CCOC(C)(CNC(c2cnns2)=O)C1 CC1(CN(C(c2ccn(CC(F)F)n2)=O)C2CC2)CCCN1C(=O)Cn1cnnn1 CC1COCC(C(=O)NCCn2cc(C(N3CCCC3C#N)=O)cn2)O1 N1(C(=O)CCc2ccc[nH]2)CCC2CCN(C(c3ncc(F)cc3F)=O)C2C1 C1(C2CCOCC2)(C(=O)NCC(CNC(c2c(C)nc(C)[nH]2)=O)O)CC1(F)F C=C(C)CCC(=O)NC1CC(C)(CNC(c2cc(C)n(C)n2)=O)C1 Cc1noc(C)c1CSCCC(=O)N(C)CCOCCNC(c1ccc(F)o1)=O C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(c2cnn(CC)c2)=O)CC(C)(C)C1 C1(NC(c2c(OC)nsc2)=O)CC(F)(F)CC1NC(=O)CC(C)F Cc1cc(C#N)ccc1C(N1CC(C(=O)NCCC2(C)CC2)CC(C)C1)=O Cc1ncc(C(=O)NCC(CO)NC(C23CC(C(F)(F)F)(C2)C3)=O)c(Cl)c1 C1(NC(c2cc(OC)nc(C)c2)=O)CC2CCC(C1)N2C(C1(S(N)(=O)=O)CC1)=O c1(CNC2CCN(C(=O)C(O)c3ccco3)C2)cc(Cl)c(Cl)cc1Cl C(CCCC(=O)NCC1CN(C(=O)C(C)SC(C)C)CC1C(F)(F)F)SC C=C(C)CN=C(NCC1(C#N)CCCC1)N1CC(OC)C(O)C1 c1(C(N2CCC(C)C(N(C(=O)C3=C(Cl)CC3)C)C2)=O)cn2ccccc2n1 c1(C(=O)NC(C2CN(C(=O)C=CS(C)(=O)=O)CCO2)C)cccc2ccn(C)c12 c1(CSCC(=O)NCCN(C(c2ccc(C)o2)=O)C)ccc(Cl)nc1 c1(NC(c2cccc(C)c2)=O)ccncc1C.C(CN)(CCOC)NC(CCC)=O N1(C(C(CC)C)=O)CCCC(N(C)C(c2ncc(OC)cn2)=O)CC1 C#Cc1ccc(C(=O)NCC2(C(=O)Nn3cncn3)CCCC2)c(C)c1 C1(CNC(Cc2cn(C)nc2)=O)CC12CCN(C(C1CC(=O)CC(=O)N1)=O)CC2 CCC(C(=O)N1CCC(CCC(=O)NCC2(Cl)CCC2)C1)N(C)C c1(C(C(=O)N(CCNC(C2CCC(=O)O2)=O)CC)(F)F)ncccc1Br c1(C(N2C(CNC(c3cnc(O)o3)=O)CC(F)C2)=O)cc2cccc(F)c2s1 CC1CCCC(CC(=O)N(CCC(=O)N(C2CCOC2)C)C2CC2)C1 c1(N2CCCC(CNC(C(c3ccc(C)cc3)C)=O)C2)ncc([N+](=O)[O-])c(C)n1 c1(CN(CCCOC)CC(=O)O)c(C)nn(-c2ccc(F)cc2)c1Cl C(=O)(C1=CS(=O)(=O)c2ccccc21)NCC1C(NC(=O)Cn2ncnn2)C1 c1(C(=O)Nc2scc(C(=O)Nc3scc(C(=O)OC)n3)n2)ccc2nccn2c1 N1(C(Cn2ncc(C)c2)=O)CCC(NC(=O)C=CCn2cncn2)C(O)C1 CC(C)C(CC1CCCC1)C(=O)NCC1CC(C)N(C(=O)CC2CCOCC2)C1 CC(CNC(C1C(CNC(=O)CC(C2CC2)C2CC2)C1(C)C)=O)CCCO c1(C(N2CCN(C(c3ccc(OC)s3)=O)CC2)=O)ccc2nsnc2c1 Cc1ccc(C(=O)N(CCC(=O)NCCF)C)o1 c1(OC)ncc(C(=O)NCC2(C)CCC(NC(C3CC(OC)C3)=O)C2)cc1Cl C(N=c1[nH]c2c(c(=NCCS(=O)(=O)CC)[nH]1)COCC2)c1c(C)c(F)ccc1 N1(C(CSCCC(C)C)=O)CC(O)CC1CNC(=O)C(C)C(F)F CC(C)(CS(C)(=O)=O)C(=O)N1CCC(CCNC(=O)C=CBr)C1 Cc1ncc(-c2nc(Cn3cc(Br)cn3)nn2-c2ccc(C(=O)O)cc2)c(O)n1 c1(CCC)nc(C(=O)N(C2CCCC2)CCNC(c2oncc2C)=O)co1 [N-]=[N+]=NC12CCC(C(=O)NC3CCCN(C(c4n[nH]c(=N)[nH]4)=O)CC3)(CC1)C2 c1(C(N(CC(C)NC(C(C)OC)=O)C)=O)ccsc1SC C(=O)(CC(C)(O)C1CC1)NC(C1C=CC(CNC(C(C)OCC2CC2)=O)C1)=O C1(CNC(c2cnc(C3CC3)[nH]2)=O)C(C2CC2)CCN1C(C1(CF)CC1)=O c1(C(N2CC3CN(Cc4ccc5cc[nH]c5n4)CC3C2)=O)cc(F)c(Br)c(F)c1 CCC(CC(=O)NOCC(C)CC)NC(=O)C=CC1CCC1 C(=O)(C1OCCc2ccccc21)NC(C)CCCC(F)(F)F C(C)(C(=O)NCCCCC1CN(C(=O)C(C)N(C)C)C1)OCC#C.C1(=O)CN1 C(=O)(C#CC1(C)CCCO1)NC1(CNC(c2ccc(C)c(Cl)c2)=O)CCOC1 C1(NC(C(Cc2cncc(Cl)c2)NC(=O)CC=C(Cl)Cl)=O)CC2(CCOC2)C1 C1(N(C)C(c2sccc2F)=O)CCC(NC(C2(C)C3COCC23)=O)CC1 Cn1cc(N)c(C(=O)NCc2ncccc2CNC(=O)Cc2ccc(F)nc2)n1 c1(SC)ccc(CCC(N2CC3CC3(CNC(c3cc(C)nn3C)=O)C2)=O)cc1 c1(CC(=O)NC(C2CCN(C(=O)COC(F)F)C2)C)nnn(C(C)(C)C)n1 N1(C(c2n(CC)ccc2)=O)CC(OC)CC1CNC(c1cncc(C)n1)=O C1(F)(CNC(c2cc(C(C)=O)on2)=O)CCN(C(c2ccc(O)nc2Cl)=O)CC1 CC1CN(C(c2cncc3[nH]ccc23)=O)CCCN1C(C1CC2C=CC1C2)=O C(=O)(C(C)CCCC(C)C)NCC(CCC)C(=O)N(CC(C)C(C)C)C N1(C(C(C2CC2)SC)=O)C2CCC1CC(C(=O)N(C)CCn1cnnc1)C2 c1(C(=O)NCc2ccc(C(=O)NC(CCCC)C)o2)cc(C)[nH]c1C N1(c2snc(C)n2)CCOC2(CCC(NC(=O)Cc3sccc3Cl)CC2)C1 C1(C(=O)NCC(N2CCN(C(c3nccc(N)c3Cl)=O)CC2)C)CCCC12CCC2 C12(NC(=O)Cc3cnc[nH]3)CCCC(CN(C(c3ccc4n[nH]cc4c3)=O)C1)C2 c1(N(C)C)nc(Cl)c(C(N2CCCCC2CNC(=O)C#CC2CC2)=O)s1 CON(Cc1ccc(C)o1)C(=O)CN(C(C1(O)CCC1)=O)CC1CC1 c1(C(=O)NCc2scc(CNC(C3(OC)CCOC3)=O)n2)scc(C)c1C.C1(C)CC1 C(=O)(C1=CCCOC1)N1CCC(CC)C1C(=O)NCc1nc(O)ccc1C N1(CC(=O)NCC2CC(C)N(C(C3CN(C(N)=O)C3)=O)C2)CCCCCC1=O C1(CC(=O)NC(CCC(=C)C)C)CCCN(C(c2ccc(NC)cc2)=O)CC1 N1(C(CCc2n(C)cnc2)=O)CC2CCCC(NC(=O)CCS(C)=O)C2C1 c1(C(=O)NC2C3CN(C(=O)Cc4cc(Cl)cs4)CC23)ccc(F)cc1Br CCCC(C(=O)N(CCC(=O)N(C)CC1CCCCC1)C)OC.C1(=O)CCCO1 C(C(C)(C)C(=O)NC12CC(NC(=O)CCc3ccsc3Br)(C1)C2)SC c1(NC(C2C(CNC(COCCOCC)=O)CC2)=O)ccc(C(C)C)cc1 C=CCC(C(=O)N(CCCNC(=O)C(C)C(=O)N(C)C)C)C(C)C C1(CC=C)(C(=O)N(CC(C)(C)CNC(c2ccnn2CC(C)C)=O)C)CCCC1 C1(NC(C(CC)C)=O)CCCN(C(C2(C(=O)OC(C)(C)C)CCCC2)=O)C1 c1(CCCCC)ccc(N(c2cnc(C)cn2)C)cc1 c1(NC(c2ccc(CC(C)C)cn2)=O)cnc(F)cc1C C(=O)(CC1=CCN(C(C2(C(F)(F)F)CC2)=O)CC1)N1C(C(=O)NC)CC1 C1(NC(c2nc(C)[nH]n2)=O)CCC2(CC1)CCN(C(C13CCCC1C3(F)F)=O)C2 C(=O)(CCCC(CC)NC(=O)CC(C)(C)C#N)N1CCCC(CC)CC1 N1(C(C(=O)NC)C2(C)CC2)CCc2cnccc2C1.C(=O)CCCC1CCCO1 Cc1cc(N)c(C(N2CC(C3CN(C(C45CCCC4C5(F)F)=O)C3)C2)=O)cc1C c1(CC)nn[nH]c1C(=O)NC1CCC1CNC(=O)CSC1CC1.c12nnnn1C2 C(=O)(C(O)C(F)(F)F)N1CCC(N(C(c2cnc(C)[nH]2)=O)CC2CC2)C1 c1(C(N(C)CC2CCCN2C(c2sccc2F)=O)=O)ccc(Cl)cc1Cl c1(C(=O)NCCCN(C(=O)C=C)CCO)c[nH]c2cc(OCCOC)ccc12.OC CC(C)C(C(=O)OCC1CCC(C2OCCO2)CC1)NS(C)(=O)=O c1(C(=O)NC(C2CCCCC2)C(C)NC(CNC(=O)NC)=O)ccnn1COC c1(-n2ccc(C)n2)ccc(C(=O)NCC2CCN(C(c3cncn3C)=O)C2)cc1 CCC(CN(C)C)CC(=O)NC1CCN(C(c2cccc(N(C)C)n2)=O)C1C c1(C(=O)Nc2cc(Cl)cc(Cl)c2Cl)csc2c1CCN(Cc1cccnc1O)C2 N1(C(c2[nH]c(C)c(C)c2C)=O)CCC2CN(C(=O)CN3CCSCC3)CC12 N1(C(c2cc(C)on2)=O)CCCC(C)C1CNC(=O)C=Cc1sccc1C c1(C(=O)NC2CN(C(c3ccc(N)c(F)c3)=O)C3C2C3)coc2c(F)cccc12 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC=CC(NC(c2ccc(C(N)=O)o2)=O)C1 C(=O)(C(CC(C)C)n1cc(S)cn1)N1C(C(C)(C)OC)CC1 N1(C(CCC(=O)OC)=O)CCC(F)(F)C(C(=O)NCc2ccc(Cl)c(F)c2)C1 c1(C(=O)NC2CCN(C(=O)CCCF)CC2)nc2ccccc2o1 C1(C(=O)NCC(CC(=O)NCCc2ncc[nH]2)O)CN2CCC1CC2 c1(-n2cc(CNC(c3c(NC)cccc3)=O)nn2)cc(C#N)cc2ccccc12 N1(C(C(COCC=C)C(C)(C)C)=O)CCC2C(C1)CN2C(=O)COc1ccsc1 C(=O)(CCC(C(C)(C)C)NC(=O)OC(=O)CC(c1cccs1)C1CCC1)OC N1(C(c2ccc(C)c(F)c2)=O)CC(NC(=O)Cc2ccn(C)n2)C2(CCC2)C1 CC1(C)CC(NC(=O)CCCC2CCOCC2)CN(c2ccc(C#N)nn2)C1 S(=O)(=O)(c1ccc(N2CC3CCC(CC3)C2)cc1Br)NC(COC)CO CN1CCN(CC(=O)NCC2CCC(NC(C3(F)CCOC3C)=O)CC2)CC1 c1(N2CCC(C(C)NC(c3c(CSC)cccn3)=O)CC2)nnccc1C#N C1(OC)CCN(C(c2ccc(CNC(=O)CC3CC3)nc2)=O)C(C)C1 C1(O)(CNC(C(C(C)O)NC(c2ccc(C)o2)=O)=O)CC2C=CC1C2 C(CNC(C1CCCS1)=O)(C(C)C(C)C)NC(c1ccnc(OC)n1)=O C#CC1COCCN1C(=O)CCCCNC(c1cc2n(n1)CCO2)=O CC1CN(C(=O)CC2CC2C(F)(F)F)CCN(C(C2CC23CCC3)=O)C1 c1(C(N(CCCNC(c2cnn(C(C)(C)C)c2)=O)C)=O)n[nH]c2ccc(Cl)cc12 C(=O)(C1=C(C)CCCC1(C)C)N1CCC(NC(C(C(CC)C)O)=O)(COC)CC1 C1(N(C(c2ccc(OC)nn2)=O)C)CCCN(C(=O)C(C)C#N)CC1 C(=O)(CCCCCN(C)C)NC(CNC(c1cnn(CCCC)c1C)=O)(C)CC c1(C(=O)NC2C(NC(C3CC(OCC)C3)=O)C2)cc2cc(F)ccc2s1 N1(C(c2c(C)[nH]c(C)c2C)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)CC1C C(N=c1ccc(Br)c(S(=O)(=O)N2CCCC(CF)C2)[nH]1)C1(CS(C)(=O)=O)CCC1 C1(CC(=O)NC2(COC)CC2)C2CCC(C2)N1C(=O)CN1CC2CC2C1 c1(NC(C2CC(=C)CN2C(c2cc(F)c(Br)cc2C)=O)=O)ccc(F)cc1C#N c1(C(=O)OC)nc(Br)ccc1NC(C1(F)CN(Cc2c(C)cccc2Br)C1)=O Cc1ccccc1COc1nc(C)n(-c2cccc(F)c2)n1.n1(C2CC2)nccn1 C1(CNC(c2ccc(C(N)=O)cn2)=O)C2CCC1CN(C(=O)CSC(F)(F)F)C2 c1(CCNC(N(C)Cc2nc(CC)on2)=O)cnc2ncccn12 N1(C(c2ccc(CC)o2)=O)CC2CCC1CN2Cc1ccccc1 C(=O)(C1=CCOCC1)N1C(C)CC(NC(C(C(C)C)NC(C)=O)=O)C1 n1(CC)ncnc1C(=O)NC1CCCC1NC(=O)CCc1ccccn1 C(=O)(C(O)C(C)(C)CC)N(C(CN(C(c1cncc(NCC)c1)=O)C)C)C c1(C(=O)OC)cn2c(CNC3CC(CNC(=O)NC(C)(C)C)C3)cnc2s1 N1(C(c2cc(C)cc(Cl)c2)=O)CCC(C2CC2)C1CNC(C1CC1F)=O N1(C(c2cc(CC)oc2C)=O)CCC(C)C(CNC(=O)CCc2n[nH]c(=N)s2)C1 C1(C2CN(C(=O)Cc3ccno3)C2)(NC(c2nc(C)sc2)=O)CC1 c1(CN(C)CCN(S(=O)(=O)CC2CCC2c2nc[nH]n2)C)ccc(F)cc1Cl Cn1nc(C(N2CCC(CCNC(c3nc(=O)n(C)[nH]3)=O)C2)=O)cc1O c1(CCCC(=O)NCC(C2CCC2)NC(=O)COC2CC2F)c(F)cccc1F Cc1nc(C)n(CCCC(=O)NCC2CCC(NC(=O)C(F)(F)CO)CC2)n1 C1(CNC(=O)Cc2cnccc2Cl)CC2(CO1)CN(C(C1CC(F)C(=O)N1)=O)C2 C1(CC)(NC(=O)CCC(C)NC=O)CCN(C(C2CCCS2)=O)CC1 CCCCCCCCC(C)C(=O)N(CCNC(=O)C(C)(C)NS(C)(=O)=O)C(C)C c1(CC(=O)NCC(CC)(C)NC(c2ccc(O)cc2C)=O)ccc2c(c1)CCO2 C1(C(=O)NC(C(=O)N(C)CC)C)CC2CC1CN(C(=O)CCC(C)N(C)C)C2 c1(CCC(N2CCC(C(C)NC(=O)CSS(C)(=O)=O)C2)=O)ccc(O)cc1 c1(CCCNC(=O)NCn2ccc(CNCc3ccccc3)n2)ccccc1Cl C(=O)(C(C#N)C(C)C)NCC(CCC)NC(c1cscc1C1CC1)=O C(N=c1cc(C(F)(F)F)nc[nH]1)C1CC(NC(CC(C)c2cccnc2)=O)C1 C1(NC(c2cc(C)cc(F)c2)=O)CN(c2ccnc3ncnn23)C2CCCCC12 c1(OC)ccc2occ(C(N3CCCN(C(c4cnco4)=O)CC3)=O)c2c1 C12(C(N3CC(NC(C4CCc5ccnn5C4)=O)C(O)C3)=O)CCC(F)(CC1)CC2 Cc1ccc(Br)c(C(N2CCC(O)C2C(=O)N(c2ccc(F)cc2C)C(C)C)=O)c1 N1(C(c2cc(CC(F)(F)F)ccc2F)C(=O)NC)CCC2(C(=O)NC)CCCC12 CC1(C)CN(C(=O)CC23CCC2CN(C(C2CCC(=O)C2)=O)C3)CC1CO c1(C(N(CCN(C(C=Cc2n(CC)ccn2)=O)C)C)=O)c(C)cc(C)oc1=O c1(N2CC(Br)=C(C)CC2)ccc(S(=O)(=O)NCC#Cc2ccc(F)cc2)cn1 C(=O)(C(CCC)C(=O)OC)N1CC(CC(N2CCC(C#CC)C2)=O)(OC)C1 N1(C(C=C(CC)C)=O)CC(C)CCC1CNC(=O)CNC(c1ncccn1)=O C1(C2CC2)(C(=O)NCCCCC#C)CN(C(=O)CC(C)N(C)C)C1 c1(NC(=O)NCc2cnc(C3(N)CC3)nc2)cc(Cl)cc(Cl)c1F N1(C(C2(C(=O)NC)CC2)=O)CC2(CCC2)CC1C(=O)NOCc1nc[nH]n1 C(C(O)CC(=O)NCC(=O)NCCC1CCCC12CC2)NC(=O)CC1CCCC1 N1(C(c2c(C)nn(CCO)c2)=O)CCN(C(C2CC2C)=O)CC1c1ccncc1 c1(-c2nc(C)c(C(=O)NCc3ccc4sncc4c3)s2)cnn2c1CN(C)CC2 C12CCN(C1CO)C2=O.C12(C(N3CCC(OC)C3)=O)CC(CN1C1CC1)C2 c1(Cn2cc(C(N(C(C3CC(C)SCC3)=O)C)C)nn2)cccc(Cl)c1F c1(CN2C(COCCCCC=C)CC2)cc(NC(=O)O)sc1Br C(=O)(C#CC1(C)CC1)N(C(CCNC(c1c(C)ncn1O)=O)C)C c1(C(=O)Nc2cn(C)c(C(=O)NCCCC(F)(F)F)n2)c[nH]c2ccc(Cl)cc12 C1(C(=O)NC(C)CNC(=O)CC(C)c2ccco2)CCN(C)C(=O)C1 C1(F)(CNC(CSC)=O)CC2CCC(C1)N2C(=O)CSCC(F)(F)F N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(=O)COCC(F)(F)F)CC1C1CC1 c1(OC)ccc(CC(N2CC(O)(C(C)NC(=O)C(C)C3CC3)C2)=O)cc1F O=c1cc(CNCc2cc(OC(F)F)cs2)on1-c1ccccc1Cl c1(NC(=O)CC2CN(C(c3ccc(=O)oc3)=O)CCO2)cnn2cccnc12 c1(C(=O)NC2CCC(N(C(=O)CCC3CC3)C)CC2)nc(Cl)c(=O)[nH]c1N c1(CSC)ccccc1C(=O)NCC(n1cc(CCS(N)(=O)=O)nn1)(C)C c1(C(=O)NC2CN(C(C=C(C)C(C)(C)C)=O)CC(O)C2)cnc2n(c1=O)CCS2 N1(C(c2c(SC)scc2)=O)CCC2(CC1)CC2CNC(C1CCNC1=O)=O CCC(C)C(O)C(C)C(=O)NC1CC(O)C1CC(=O)NCc1nc(C)no1 C1(C(=O)NC2CC2)CC(CNC(=O)CN2CC=CC2)CC1O.N12CC(C1)C2=O c1(CNC(C(n2cc(-c3ccc(C)nc3)nn2)C)=O)cnc2sccn12 C(=O)(C(CC(C)SC)N1CCCC(O)(c2ccccc2)C1)NCC C1(NC(C(C2CC2)SC)=O)CCC(C)(NC(c2cc(COC)cs2)=O)CC1 CCC(C)CCC(=O)NCC(O)CNC(c1c(-c2ccccc2F)noc1C)=O C1(CC=C)(NC(=O)C(F)(F)CC2CCCO2)CCN(C(=O)Cc2ccsn2)C1 N1(C(=O)OCC)CSCC1C(=O)NC1CN(C(=O)CN2CC3CC3C2)C1 Cc1ccc(CN(CCC(=O)N(C)CCN(C(=O)C(C(C)C)N(C)C)C)C)cc1 Cn1cccc1C=CC(=O)NC1(CNC(C2CC(C#N)C2)=O)CCOC1 CC12CN(C(=O)CC3(O)CCOC3)C(C(=O)NC3CCC3c3ccccc3)(C1)C2 C(=O)(C(C)(C)CC(=O)NC1CCC1CNC(c1ccnc(N(C)C)c1)=O)OCC C(=O)(C1CCCc2sc(C)nc21)NCC(CCOC)NC(=O)Cc1ccccc1 C1(C(=O)NCC2CCC(=O)N2)CC(F)CN1C(=O)C1CC1 n1(CC(=O)NCCCN(C(CC=C)=O)C)nc2n(c(=O)c1=O)CCOC2 C(C#Cc1cccnc1)NC(CCC1CCCN(C(c2cnc(OC)s2)=O)C1)=O CC1CC(NC(=O)NCCc2ccc(N)cc2)CC(C)C1 C1(C(=O)OC)C2CC3C(C2NCC(CC2CN(C(c4ncn(C)n4)=O)C2)(C)O)C13 c1(C(=O)NC(C2CC(NC(C3CC3(C)C(F)F)=O)C2)C)cn2cc[nH]c(=O)c2n1 N1(C(CSCC(N)=O)=O)CCC(NC(=O)C2=NOC(C(C)(C)C)C2)C(F)C1 C(C(C)(C)CC(=O)N1CC2C(NC(C3CCCN3C)=O)C2C1)N(C)C C(CC(=O)N(CC(C)O)C)N(C(=O)CNC(C1CC1C)=O)CC C=CC(C)(C)C(=O)NCC(O)CCNC(c1cc(-c2ccc(F)cc2)n(C)n1)=O c1(N(CC(=O)NCCN(C(C2CC2(F)Cl)=O)CC)C)ccnc(Cl)n1 C(C(O)C(F)(F)F)NC(CC1N(C(CCn2c(C)ncc2)=O)CC1)=O c1(OCC(=O)N(CC(C)NC(C(=O)NC(C)C)=O)C)ccc(F)cc1 Cc1c(C)c(C)c(C(=O)NCC(F)CNC(c2cnc3n2CCC3)=O)c(C)c1C c1(OC)cccc(C(N2CC(NC(c3ccc(C(F)F)cc3)=O)C3CC23)=O)c1N C1(C)(CC(=O)NC(C2(CNC(=O)CC(C)c3ccco3)CC2)C)CCCO1 Cn1ccnc1CCC(=O)NCCCNC(C1CCC1(F)F)=O C(=O)(C1COc2ccccc21)N1CCCC(O)(CNC(=O)CS(=O)(=O)C2CC2)C1 Cc1ccc(S(=O)(=O)N2CCN(C(=O)C(F)CC3CC(F)(F)C3)CC2)s1 Cc1cc(N2CCC(C(F)(F)F)(C(N3CCC4CCCC34)=O)CC2)nc(C#N)c1 C1(NC(C2N(CCC)CCC2)=O)(CO)CCCN(C(=O)C(C)(C)O)C1 C1(C(N(CCN(C(C(COC)OC)=O)C)C)=O)CCc2ccccc2N1 Cc1ccc(C(N2CCCCC2CCCNC(C2(C)CC=CCO2)=O)=O)c(C)c1 NS(=O)(=O)c1cc(NC(=O)CC(=O)CCc2ccc(O)c(O)c2)ccc1Cl c1(C(c2ccccc2)NCc2c(C)cc(C)s2)cc(Br)ccc1Br C12CC3CCC(C1)N3C2=O.Nc1cc(Cl)ccc1-c1nn[nH]n1.c12oc-1cc2O S(=O)(=O)(c1ccc(C(C)=O)cc1)N(C(c1cccc(OC)c1)C)C C(N=C(NCC1CC1)NCC1CC2CC1C2)C1CCN(C(C)(C)C)C1 C1(NC(CCC(=O)NCCC)=O)CC2CC(NC(C3CC(C)(C)C3)=O)C1C2 Cn1nc(Br)cc1CC(=O)NCCCC(N1CC(C2CCCCC2)C1)=O N1(C(CCCC)C(=O)NC)CC(CC)OC(CC)C1(C)C N1(C(CCn2ncc(C)c2)=O)CC(=O)NCC1C(=O)NCc1ccc(F)cc1O C1(CNC(CN2CC(CC)C2)=O)CN(C(c2ccnn2CCF)=O)CC1C c1(OC)ccc(C(=O)NC2CC(NC(C3CCCN(C)C3)=O)C2)cc1OC(F)F N1(CCS(=O)(=O)N(C)C)CCC(O)(C(N2CC(C(=O)OC)C(C(=O)O)C2)=O)CC1 C1(C(=O)NC2CCN(C(c3c(C(C)C)ccs3)=O)C2)CCCC1C1CC1 c12nc(n(Cc3cncnc3)n1)-c1c[nH]c(c1)CCNC2C.CCSC N1(C(C(C)(N(C)C(c2cscn2)=O)C2CC2)=O)CCOC(C2(C)CC2)C1 C1(C(C)NC(=O)COCC(C)(C)C)CCCCCN1C(c1ccn(CCF)n1)=O Cc1ccncc1C(=O)NC(CCF)C(=O)NCC(C)S(N)(=O)=O CC(C(=O)N(CC(=O)O)CC(C)C)C1CCCN1 c1(CNc2nccc(-c3ccc(C(C)(C)O)cc3)c2)cc(I)ccc1[N+](=O)[O-] C(=O)(C1=NOC2(CCC2)C1)NCC(C)CN(C)C(C1CCN(C)C(=O)C1)=O c1(CCC)ccc(N)c(C(N2CCN(C(C3CC(C)(F)C3)=O)CC2)=O)c1 C1(CC)(NC(=O)C(c2ccc(F)cc2)C)CCN(C(=O)CCCN=[N+]=[N-])CC1 C1(NC(=O)Cn2nccn2)CCCN(C(c2cc(F)cc3nc[nH]c23)=O)CC1F C(=O)(C(O)CN1CCCC1)NC(C1CN(C(=O)C(Cl)=CCl)C1)C C1(NC(c2c(C)n(C3CC3)cc2)=O)CCC2(CC1)CN(C(=O)C=CCO)CCO2 c1(C2(C(C3(N)CC(C)SC3)c3n(CC=C)nnn3)CC2)cccc(C)n1 N1(C(c2c[nH]c(=NC)o2)=O)C2CCC1CC(NC(=O)C=CS(=O)(=O)CC)C2 c1(CN(C)C)ccc(C(=O)NCC2(NC(C(CC)C)=O)CC2)cc1 CCCCCCC(C)C(=O)NC(C)CNC(c1cnc2c(c1)CCC2)=O c1(C(=O)NC(c2ccc(CC)cc2)C#N)cc(-n2cnnn2)ccc1Cl C1(O)(CNC(=O)C(F)=CC2CC2)CC(C(=O)NC2(C3CCCCO3)CC2)C1 CNS(=O)(=O)N1CCC(C(=O)NC23CC2CN(C(=O)CS(N)(=O)=O)C3)CC1 C(CC(C(C)C)N(C)C)N(C(c1n(CC)ccc1)=O)C.C1(F)(C=O)CCOCC1 N1(C(C(C)(C)N(C)C)=O)CCC(O)(CNC(c2ccccc2CO)=O)C1 C1(CC(N2CC(OC)C2)=O)C2CCCC2N1C(C1CC1C1CCCC1)=O c1(C(CC(=O)NC(C2(CNC(=O)C3=CCSC3)CC2)C)C)c[nH]c2ccccc12 C(=O)(CCC(F)(F)Cn1cc(C2CCOC2)nn1)NC(c1ccc(F)cc1)C CC1=C(C)CC(NC(=O)C(=O)NCc2csc(N)n2)CC1.c1(C=O)c(C)ccn1C c1(CCCC(=O)NC2CCC2NC(=O)C(F)=C2CCCC2)ccc(Br)cn1 N1(C(CC2CCC(C)(C)CC2)=O)CCCCC2(CCN(c3ccnc(Cl)n3)C2)C1 N1(C(CC2CC(NC(c3c(CC)cno3)=O)C2(C)C)=O)CC2CCCCC12C c1(CCC(=O)NC2CC(Cn3cc(CCNS(C)(=O)=O)nn3)C2)ccccc1Cl C(=O)(CCCC(=O)NCCCOCCCNC(=O)CC1CC1C1CC1)OCC.OCC c1(CC(N2CC(C)(NC(CN(C)C(C3CC3)C3CC3)=O)C2)=O)c(Br)cnn1C C1(NC(=O)Cn2cnnn2)(CO)CCCN(C(=O)CCc2cccnc2F)C1 N1(C(=O)CCOCC(F)F)CCN(C(c2cc(Cl)ncc2O)=O)C(CF)C1 C(=O)(C1CCCc2nn[nH]c21)N1CC(C)(NC(=O)COC2(C)CCC2)C1 c1(C(=O)NCCN(C(C(CCC)(C)O)=O)C)nc2c(Br)cccn2c1N Cc1cccc(C(=O)NC2CC(C(=O)N(C)Cc3ccccc3)C2)c1O CCC1=C(C(=O)N2CC3CC2C3C(=O)NC2CC(=O)N(C)C2=O)CCCO1 Cc1c(C(N2CCOCC2CNC(C2CN(C)C2)=O)=O)cc(N)cc1O CC(C)(CF)C(=O)N1CCCC(C(=O)NCCNC(C2CCCOC2)=O)C1 C1(C(N(CC)CC2CCCN2C(=O)C(C2CC2)C2CC2)=O)C2(CCC2)C12CCC2 c1(CC(=O)NC2C(NC(C=CC)=O)CCCCC2)ccccc1S(C)=O C1(c2cn(C(C(=O)NC(CC(C)C)(C)C)C)nn2)CCc2nccn21 C1(C(N2CC=C(CNC(CCNS(CC)(=O)=O)=O)CC2)=O)Cc2ccccc2S1 C1(C2CCCN(C(c3ccccc3F)=O)C2)(NC(C2CNC(=O)N2)=O)CC1 N1(Cc2c(=O)c3ccc(C)cc3[nH]c2)CC=C(c2cccc(Br)c2)CC1 C1(C(N2C3(C(=O)NCC(C4CCC4)OCC)CC3CC2)=O)CCC(C2CC2)C1 C(=O)(CCC(CF)CF)NC1(C(=O)NCC(c2ccccn2)O)C(C)(C)C1 C1(NC(C(C)(C)C)=O)COC2CN(C(c3ccnn3CC3CC3)=O)CC12 c1(C(=O)NCC2(F)CC(CNC(C(C(C)C)OCC)=O)C2)cnc2n1CCCC2 C(C(C(F)(F)F)OC)NC(CC1C(C(=O)C(C)=O)C1)=O.C(C(C)(C)O)SC.C(C=O)N c1(OC)cc(Br)cc(NC(C2CCC(NC(=O)C=CC3CC3)CC2)=O)n1 C1(NC(C(C(C)C)F)=O)CCCN(C(c2ncccn2)=O)CC1 C(=O)(C(C(=O)NCC1CCN1C(c1ccc(-c2ccncc2)o1)=O)OC)OC N1(C(c2ncn(CC)c2)=O)CCC(C(=O)N(C(C)CSC)C)C1C c1(C(c2ccccc2)C(=O)NC(C(=O)OC)C2(O)CCC2)cccnc1 C(=O)(CC(C)C(F)(F)C(F)(F)F)NC(CC)(CNC(=O)Cc1conc1C)CC N1(C(C(CC)=CC)=O)CC2CCC(CNC(c3ncccc3SC)=O)C2C1 c1(C(N2CCC(C)(NC(CC3CCC(C)(C)C3)=O)C2)=O)cncc2ncccc12 Cc1ccc(C=CC(=O)NCCC2CN(C(=O)CC3CC3C)CCO2)o1 C1(CCC(=O)NC(CC=C)CNC(C2(c3ccn(C)n3)CC2)=O)CCN(C)CC1 C(C(CCC)C(=O)N1CCCC(C)(N(C)C)C1)NC(C=CCOC)=O n1(CC(=O)NC(Cc2ccoc2)CO)cc(-c2ccccc2)nn1 C1(C(=O)NCCN(C(=O)C=CBr)CC)Cc2ccc(F)cc2O1 C1(C(N2CC(NC(c3cc(Cl)c(F)cc3F)=O)C2)=O)CCc2nc(O)[nH]c2C1 c1(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)C)csc2c(F)cccc12 c1(C(=O)NC(CN(C(c2cc(C)nnc2)=O)C)C)nc2sccn2c1C C1(NC(C2CC3C=CC2O3)=O)CN(C(=O)CN2CSCC2=O)CC12CC2 Cc1ccc(C(=O)NCCCCCCNC(C23CSCC2C3(F)F)=O)c(O)n1 N1(C(C=C(CCC)C)=O)CCN(C(=O)C=CC(C)C)C2COCC12 C1(C(=O)NC(CCC)C2CCC2)CN(C(=O)C(C)=C(C)C)CC12CC2 c1(OC)coc(C(=O)NCC(C)(C2CC2)NC(=O)C2=CCOC2)cc1=O N(C1CCS(=O)(=O)c2ccc(F)cc21)C(C12CCC(CC1O)C2)=O N1(S(CN(C(C)=O)CC2COc3ccccc3O2)(=O)=O)CCC2(C1)OCC1CC21 c1(C(=O)NC23CC(Nc4nnccc4C(F)(F)F)(C2)C3)c(F)ccc(Cl)c1Cl CC(C)C(C)C(CNC(=O)Cn1ccc(O)nc1=O)NC(C1(F)CC1)=O c1(-c2ccc(C3CC(CC)OCC3)cc2)ccc(S(=O)(=O)N2CCCCC2)cc1 N1(C(C(C(C)C)NC=O)=O)CCN(C(C2CCN(C)C2)=O)C(C(C)C)C1 N1(C(C2CC23CCOCC3)C(=O)OCC)CCC(C)(F)CC1.C12(CC1)CC(=O)N2 N1(C(C2OCC(C)(C)C2)=O)CCC2(CCC2)C(NC(c2ccc(F)c(Cl)n2)=O)C1 CCS(=O)(=O)CC(=O)N(CC(C)O)CCOCC1CN(C(C)=O)C1 c1(NC(C=CCN(C)C(C2CC2(F)Cl)=O)=O)ccc(Cl)c(O)c1 C(C(O)C(=O)NCC1CCCC1CNC(C1(c2ccncc2)CC1)=O)N(C)C CCC(CC(=O)NCC1C(C)CCN1C(c1ccncc1Cl)=O)CC(F)(F)F c1(C(=O)NC(CC#C)Cc2ccccc2)cc2scc(Cl)c2s1 c1(N2CCCC(C(=O)NCc3ccnc(SC)n3)C2)cc(C(F)(F)F)nc(C)n1 C(c1cccc(C)c1)=CC(N1CCC(OCCNC(C(COC)O)=O)C1)=O N1(C(C2CN(C(C)=O)C2)=O)CCCCC1C(C)(C)C(=O)NCc1ccc(C)cn1 c1(C(=O)NCC(CNC(COC2(C)CCCC2)=O)O)cc2n(n1)CCCO2 c1(CC)ccc(NC(=O)C(C2CCCC2(C)C)N(C2CC2)CC)cc1.C1C(=O)O1 Cn1cc(Cl)c(CC(=O)NC2(CO)CN(C(=O)Cc3cncnc3O)C2)n1 CN1CCN(C(=O)C(F)(F)c2sccc2Cl)CC1C(=O)OC(C)(C)C S(=O)(=O)(c1ccc2scnc2c1)Nc1cccc(C(C(=O)OCC)(F)F)c1 N1(C(COC)=O)CCN(C(C2CCS2(=O)=O)=O)CC1c1nccn1C [N-]=[N+]=NC1CC(C(=O)NOCc2ccsc2)N(C(C2CC3CCCC3C2)=O)C1 N1(C(c2c(C)ccc(F)c2)=O)CCOC2(CCN(S(=O)(=O)C(F)(F)F)CC2)C1 C1(CCCCNC(CCCOC)=O)CCN(C(=O)CC2CCCOC2C)CC1 c1(SC)cnc(F)c(C(=O)Nc2ccnc(F)c2C)c1 CCC(CC)(CC)C(=O)N1CCOC(C(N2CC(O)(CCO)C2)=O)C1 c1(OC)ccc(Cl)c(C(=O)NC2CC(C)(NC(=O)CCCNC(N)=O)C2)c1F O=C(CCCn1cccn1)NC1(CCNC(C2(F)CCOC2)=O)CCCC1 c1(C(N2CC(NC(c3c(C)nn[nH]3)=O)C2)=O)cnn2c(-c3cccs3)ccnc12 c1(C(=O)NCC2(NC(C(C)NS(C)(=O)=O)=O)CCOC2)nccc(N)c1Cl C1(NC(C(C)CC2CC2)=O)CCCCN(C(c2cnn(C)c2Cl)=O)C1 C(=O)(CCCCC(F)(F)F)NC1CCCCCN(C(C2N(CCC)CCC2)=O)C1 CCN=C(NCCC(N1CCOCC1)C)NCC1CCOC1(C)C Cc1cc(CCC(=O)N(C(C)CN(C)C(c2ccc(Cl)[nH]2)=O)C)ccc1Cl c1(C(N2CCC(NC(CCN(CCC)C)=O)CC2C)=O)c[nH]c2cnccc12 c1(SCC(=O)N(C(C)C)CCN(C)C(C2CCOC2)=O)cc(F)ccc1F C1(NC(=O)CCSc2ccncc2)CC12CCC(NC(C1CC=CC1)=O)CC2 N1(CC2CCC(F)CC2)CCN(C(C2(N(C)C(=O)C3CC3)CC2)=O)CC1 C1(CC)CCC(C)CN1C(c1cn(C(C)(C)C)nc1C(=O)O)=O c1(C(N2CCCC2c2cncn2C2CC2)=O)cc(Cl)c([N+](=O)[O-])cc1Cl n1(C(C(=O)NCC)C2CCOC2)cc(CN(CCO)CC)nn1.CCC1CO1.CC C1(C(=O)NCCCNC(CCc2n(C)cnc2)=O)CCCCS1(=O)=O c1(CC(=O)NC2C(NC(C(CC=CCC)C)=O)CCCC2)ccc(C#N)nc1 O(N=C1CCCCCC1)CC(=O)NC1C(C)CN(C(c2cc(CF)on2)=O)CC1 N1(c2nnc(C)n2S(=O)(=O)c2cccnc2F)CCC(C)C2(CCCCC2)C1 c1(CC(=O)NC2C(F)CCN(C(CC(CC)C)=O)C2)cccc2c1OCCO2 c1(C(=O)NCC2CN(C(c3ccc(Br)o3)=O)C3CC23)cc2sccc2cn1 c1(CC)nc(C)c(CNC(C2CCCN2C(C2(CF)CC(=O)C2)=O)=O)o1 c1(C(CC)C)ccc(C(=O)NC(C)CC2CCN(C(=O)C(F)F)CC2)cc1 C(=O)(CC(C)CC(F)(F)F)N(C(CNC(c1cc(C)c(F)cc1F)=O)C1CC1)C c1(C(N(C(CCNC(CCCOC(C)C)=O)C)C)=O)ccncc1N C1(OC)CCCO1.C12(CC1)CN(C)C(=O)COCC(=O)N2.C1(CO)CC1 N1(c2ccc(C)nc2Cl)C2CCC1CN(C(c1cc(C3CC3)on1)=O)C2 Cc1ccn2ncc(C(=O)NC3CCC(NC(C4CN(C)CC4C)=O)CC3)c2n1 CC1(C(N2CCOCC2)=O)CN(C(C2CCS2(=O)=O)=O)C1 C1(C(=O)NCCCC(C)NC(C2(C)CCOC(C)C2)=O)CCCCC(=O)C1 N1(C(c2c(CC)nc(C)o2)=O)CCC(C2CCN(C(C3(C)CCC3)=O)CC2)CC1 N1(C(C(C(=O)OC)OC)=O)CC2(CCCC2NC(=O)CCC=CC(C)C)C1 N1(C(c2cc(CC)no2)=O)CC(NC(=O)C(C)NC(=O)NC)C(C)C1 Cc1cc(C(N2CC(F)(F)CC2C(=O)Nc2cncc(C#N)n2)=O)cc(C)n1 Cn1nc(C(=O)NC2CCCCN(C(c3n[nH]c(O)n3)=O)C2)c2c1CCC2 C1(NC(C2C(C)(C)C2C#N)=O)C2CC3C1C3C2C(N1CCC(CN=[N+]=[N-])CC1)=O c1(C(=O)NC2(CNC(c3ccc(OC)s3)=O)CCCC2)cccn(C)c1=O CCCCC(C)C(=O)N(C)Cc1ccc(CNC(C2CC2C2CC2)=O)cc1 CCC(C(=O)Nc1c(=O)cc(C(N2CC(OCC)C2)=O)oc1)C(C)(C)CC C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(C)NC(=O)CNC(=O)C1CC1 c1(CC)nc(Cl)nc(N2CCC(C3CC3)C2CNC(C2CCCC2OC)=O)c1Cl C(C)(CS(C)=O)N(CC(CC)OCC)C(CN(C(CC)=O)C)=O C(=O)(CC1=CCOCC1)NCC1CN(C(c2cc(C(C)C)[nH]n2)=O)CC1(F)CO C12(C(N3CC(C)(CCC(=O)NCCN(C)CCO)C3)=O)C(=O)C3CC1C2C3 CCC(CC(=O)NC1CC(NC(c2sccc2OC(F)F)=O)C1)CC(F)(F)F c1(C(N(CCCNC(=O)C(C)SC(C)C)C(C)C)=O)csc2nccn12 c1(C(=O)NC2CCC(CNC(C(c3cnccn3)C)=O)C2)ccnnc1O c1(C(=O)NC2(CF)CCN(C(C34CCCC3C4)=O)C2)cnn2c1CCCC2 C1(CC(=O)NC)CN(C(C2(C)COC2)=O)CCN1C(C1CCOC1C1CC1)=O N1(C(COCc2c(C)cco2)=O)CC2(C1)SCCC2NC(C1CC2COCC2C1)=O C(=O)(C#CC1CCCO1)NCC1(CNC(C2(C#N)CCC2)=O)CCC1 c1(N(C(CCNC(=O)CN2CCCCC2)=O)CC(=O)Nc2ccoc2)ccccc1 C(=O)(C(CC1CCCC1)NC(=O)C=Cc1csnn1)NCC1CC(SC)C1 c1(C(N2C(C3(NC(CC(C)SC)=O)CC3)CCCC2)=O)nccc2[nH]ccc12 c1(C(N(CCC(C)NC(C2CC(F)C2)=O)C)=O)cc(F)c(F)c(F)c1N N1(C(Cc2c(C)non2)=O)CC2(CCCC2)C1C(=O)NC1CC(=C2CC2)C1 C1(OC)CCC(C(=O)NCC(C2CC2)NC(C2CC2CC(C)(C)C)=O)CC1 c1(CNC(C(n2c(C)ncc2)C)=O)cccc(C(N2CCCC(C(C)C)C2)=O)n1 C1(CN(C(=O)CCCC2(NC(C3CC(F)(F)CS3)=O)CCC2)C)CC2(CC2)CO1 N1(S(=O)(=O)CC2CC2)CC2CCC(C1)N(C(=O)CC1CCC1)C2 c1(CNC(=NCCOCC)NCc2csnn2)cc(Br)ccc1F C(=O)(C(C)NC(C1CCC1)=O)N(CC(C)N(C(COC(CC)C)=O)C)C C(S(C)(=O)=O)CCN(CCCN)C(C1(C(F)F)CC1)=O.C1(C)(C(=O)OC)CC1 c1(C(=O)NC23CCN(C(=O)C4=COCCC4)CC2C3)nccc2ncccc12 C1(N(C(C(C2CC2)OC)=O)C)CCC(NC(=O)CCN2CCCCC2)CC1 C1(C(=O)NCCC2CC2)CCCC12CCN(Cc1ccc(F)cc1)C2 c1(-c2c(C)cccc2)cc(=NC(=O)C(=O)N2CC3OCC(CO)C3C2)[nH][nH]1 c1(C(N2CCC(=C)CC2C(=O)NC2CC3CCC2O3)=O)nccc2[nH]ccc12 N1(C(C2ON=C(C)C2)=O)CCCN(C(=O)CCC2CCC(=O)N2)CCC1 Nc1cc(C(=O)NCc2cn(CC(=O)NCCN3CC4CC4C3)nn2)cc(F)c1 Cc1ccc(C=CC(=O)NC2CC(=CC(=O)N(C)CC3CC3)C2)cc1 C(C(C)(C)CC(=O)NC1CCCC1NC(c1ccc(C(F)(F)F)c(O)c1)=O)OC C(c1ccccc1[N+](=O)[O-])=CC(=O)NCCC1CN(C(C2CCS(=O)(=O)N2)=O)C1 C1(C(=O)NCC2CCCCC2Nc2ncnc(Cl)c2F)C2CCCCCCC12 C=CC(C)(CC)C(=O)NCC(C(C)(C)C)NC(c1ccc(=O)n(CC(C)O)c1)=O C1(NC(c2nc(OC)cc(OC)n2)=O)CCCCCC1NC(c1cc(Cl)no1)=O C(=O)(C1(C)Cc2cccc(Cl)c21)N1CCCC(C)(NC(c2cc(C)oc2)=O)C1 C1(C(=O)NC2CC3(CCN(C(=O)C4=COCC4)C3)C2)CC2(CCCCC2)S1(=O)=O S(=O)(=O)(c1cccnc1N)N.c1(CN(CC(n2cccn2)C)C)cc(Cl)ccc1F N1(C(c2c(OC)n[nH]c2)=O)CC2CC1CN2C(c1cc(C(F)F)cs1)=O C1(C(N2C(CCNC(C3N(S(C)(=O)=O)CCC3)=O)CCC2)=O)CCC2CC2C1 c1(C(=O)OCCOCCOCCOCC#C)nn(C(C)(C)C)cc1Cl.OCC C1(C(=O)NCCCOCC)CC(C)(C)CCN1C(=O)Cc1cscn1 C(C)(CC1=CCCCC1)NC(C1(F)CCN(C(c2cc(SC)oc2)=O)C1)=O N1(C(C(C)NC(N)=O)=O)CCOC(CN(C)C(C2CCSCC2)=O)C1 C12(C(=O)NCC3C(NC(C4C(C)(C)C4)=O)CCC3)CC(C)(C1)OC21CCC1 c1(C(=O)Nc2nc(C)c(C(=O)O)s2)nccc2ncncc12 c1(N(CCCNC(C=C(C)Cl)=O)C2CC2)nnc(C)c(C)n1 N1(C(C(=O)NCC)=O)CCN(CC)C(=O)C1CCCN1C(CN)CCC1CC C1(CC=C)(C(=O)NC2CCN(C(C3CCCCO3)=O)C2C)CCOCC1 Cc1[nH][nH]c(=NC(=O)C2C=CCN2C(=O)Nc2ccccn2)c1Br c1(C(=O)NC2C(CNC(c3c(C)ccc(C)c3)=O)C2)c(Cl)ccc2ccncc12 c1(OCC(=O)NCC(C)NC(=O)CCC2CCCOC2)ccc2c(c1)CCC2=O c1(C(=O)NC2CC(CNC(C(C(C)O)C)=O)C2)cnc(O)nc1O C(N=c1[nH]nc(C(F)F)s1)CC1CN(C(c2c(CC)ocn2)=O)C1 c1(OC)ccc(C(=O)NC2CN(C(C3(N(C)C)CC3)=O)CC2C)c(F)c1F N1(C(=O)Nc2cccc(C#CC)c2)CCOCC12CNC(=O)OC2 C1(CNC(=O)CCNc2ccccn2)CC(NC(=O)C(=O)NC2CC2)C12CCC2 C#CCC(C(=O)N(CCc1scnc1C1CC1)CCOCCO)CCOC.C(N)(=O)N C(C)(CCCCNC(=O)C(C)Sc1nncn1C)NC(CCc1scc(C)n1)=O C1(C(N(CCNC(=O)CC2CCSCC2)C2CC2)=O)CC2(CCC2)CO1 CC(C)C(C(=O)N1CC(N(C)C)C(CNC(c2nc3ncccn3n2)=O)C1)C(C)C Cc1ccc(F)c(OCC(=O)NCC(C)(C)CNC(C2(CN(C)C)CC2)=O)c1 Cc1c(C(N2CCN(C(C3CCSC3)=O)CC2C2CC2)=O)cccc1F Cc1ccc(F)c(CC(N2CC(OCCNC(c3ccc(Cl)nc3)=O)C2)=O)c1 n1(CC)nnc2cc(C(=O)NC(CNC(=O)C(C)O)C(C)(C)C)ccc12 N1(C(CCC(CC)OC)=O)CCC(C2CC2)(NC(c2n[nH]c3cccnc23)=O)C1 O=C1NC(=O)C2(CC(CN(c3cccc([N+](=O)[O-])c3)c3ccc(F)cc3)C2)N1 c1(NC(C2(C)CN(C(C3C(OC)CCC3)=O)C2)=O)cccc(C)c1C c1(C(N2CCC(O)(C(C)NC(C(CCC)C)=O)CC2)=O)nc2ncccn2n1 c1(C(N(C(C2N(C(CCCCCC)=O)CCC2)C2CC2)CC)=O)cnn2cccc2c1 Cc1cccc(C(=O)NCC2C=CC(NC(C3C(C)C3C)=O)C2)c1 C(=O)(CCC(C)N(C)C)NC(C)CC1CN(C(C2CN(C3CCOCC3)C2)=O)C1 c1(C(=O)NC2CCN(C(C(COC)O)=O)C2)cc(C)nc(C)n1 Cc1c(Cl)c(CNC(=NCc2conc2C(F)(F)F)NCC2CCCO2)nn1C C1(CNC(C2C(COC)(CC)C2)=O)CN(C(=O)C(c2cccn2C)=O)CC(C)(C)O1 C12(CC(N3C(CNC(C4N(CC)CCC4)=O)CC3)=O)CC3CC(CC(C3)C1)C2 C1(N(C(=O)CN2CCC(C)C2)CC)CCCN(C(=O)CCn2c(C)ccc2C)C1 C(=O)(C(C)(O)COC)N1CCC(n2cc(CCCC(CC)=O)nn2)C1 N1(C(Cc2cn(CC)nc2)=O)CC(NC(C2COC(C)C2)=O)CC2(CC2)C1 C1(NC(CN(CC)CC)=O)CC2CCC1CN2C(=O)CC1CCOC1 CN1CCCC(c2cn(CC3C=CCN3C(c3cnc[nH]3)=O)nn2)C1 c1(C(N(C(C)CN(C(=O)C(F)n2ccnc2)C)C)=O)cccc(F)c1F C1(C(=O)Nc2c(Br)c(C)n(C)n2)CCCC12CCN(Cc1cc(F)ccc1Br)C2 c1(C(=O)NCCC(C)NC(c2c(SCC)nccn2)=O)cc(C)cnc1Cl N(C1COc2ccccc21)C(C1N(C(c2c(C)nns2)=O)CC2CCC21)=O c1(C(N2C(CN(C(C(F)=CCC)=O)C3CC3)CCC2)=O)c(CC)nc(SC)nc1C CCCCC(CC)C(=O)NC1CN(C(=O)C(O)C(C(C)C)OC)CC1F N1(C(C=C(COC)C)=O)CCC2(CCN(C(C3C4CCC(C4)C3C)=O)CC2)C1 c1(CC(N2CCN(C(C(CC#C)C)=O)CC2C(F)F)=O)cccc2ccccc12 c1(CNC(C2(C)CCCO2)=O)cc(C(N2CC3CC3(CO)C2)=O)ccn1 N1(C(C(C)NC(=O)NC)=O)CCCC(F)(CNC(=O)Cc2c(C)noc2Cl)CC1 c1(C(N(C(C(n2cc(SCCCC)nn2)C)=O)C)C)ccc(C)cc1 C1(NC(C(C(C)c2ccccc2)O)=O)CN(C(c2ncc[nH]2)=O)CC2(CCC2)C1 N1(C(CCC#C)=O)CCC(NC(c2cc(O)c3ccccc3n2)=O)C(F)(F)CC1 C1(CCN(C(C2CC2C)=O)CC)CCN(C(=O)CCN(C)C(=O)OC(C)(C)C)C1 C1(C(=O)NCC(C)N(C)C(c2cnc(Br)s2)=O)CC2(CCC2O)C1 c1(C(=O)NCC(CCOC)NC(=O)Cc2cccs2)cnn(CCO)c1C(C)C C1(COC)CN(C(c2cnc(C)c(N)c2)=O)CCN1C(=O)C=CC1CCCCC1 c1(CC(=O)NC(C(CO)NC(CN(CCOC)C)=O)C)ccc(OC(C)C)cc1 Cc1ccc(C)n1NC(=O)C1CCCC(C)(C)C1NCCCN(C)C C(N=c1cc(Nc2cccnn2)nc(C)[nH]1)C1CCCC(CC)C1 CCCCC(CC)CC(=O)NC(c1ccccc1)Cc1cccc([N+](=O)[O-])c1F c1(C(N(CC(C)NC(C2(C(C)C)CCC2)=O)C)=O)ccnn1CCC(F)(F)F C(=O)(C1=CC2C=CC1C2)NCCSCC(=O)NC1CC(C)(C)C1O c1(C(=O)NC(C)CCN(C(=O)C(C)(C)c2cnco2)C)n[nH]c2c1CCCCC2 C1(C(N2CCC(NC(=O)C(O)(C3CC3)C3CC3)C2)=O)COc2ccc(Cl)cc2O1 Cc1ccc(CCC(=O)NC2CCN(C(C3CCCC4CC34)=O)C2C)cc1Br Cc1cccc(C(=O)NCC(O)CNC(C2CCC(=O)N2C)=O)c1-n1cccc1 Cc1nc(=N)[nH]c(=NCC2CN(C(C3CC(=O)N(C4CC4)C3)=O)CCO2)[nH]1 N1(C(N2CCC(CN(C)Cc3[nH]nc(CC)n3)CC2)=O)CCC2(CCSC2)C1 c1(C(N2CC(C(C)(C)O)(CNC(C(C)(C)O)=O)C2)=O)ccn2c1CS(=O)(=O)CC2 Cn1cc(C2(C(=O)NCC3CCC3(C)C)CC2)cn1.C12CC1CNC2=O c1(C(N2CC(OC)C(C(=O)O)C2)=O)ccnc2c(Cl)c(C)ccc12 Cc1cnc(C(=O)NC2CC(F)(CNC(=O)C(C)C(C)(C)C)C2)cc1Br c1(CC)ccnc(C(N2CCCCC2CN(C(=O)Cc2cn[nH]c2)CC)=O)c1 O=C1CN(C2CCC(NC(=O)COc3ccccc3Cl)CC2)CCN1 C1(CC(=O)NC(CC)CN(C(=O)CCc2cnc[nH]2)CC)CC2CCC1C2 c1(C(=O)NCC(CCNC(CSCCC)=O)O)ccncc1OC c1(SC)nc(O)nc(C)c1C(=O)NCC(CNC(c1ccnnc1S)=O)OC Cn1ccc2[nH]c(C(=O)NC3CCCN(C(=O)C(Cl)=CCl)CC3)cc12 N1(C(c2c(C)cco2)=O)CCC(O)(CNC(C2CCCN2C)=O)C1 C1(C)(NC(c2ccc(CNC(C3C(OC)CC3)=O)nc2)=O)CCCCC1(C)C N1(C(c2c(CC)occ2)=O)CCC2(CC1)CC(C)N(C(c1ccncc1O)=O)C2 C(=O)(C(O)CC1CCOCC1)N(C(C)CNC(c1nncs1)=O)CC c1(CC(C)C)ccc(CC(=O)NCC2CN(C(c3cnccn3)=O)C3CC23)cc1 C1(OC)CN(C(C2(Br)CC2)=O)CC1NC(c1ccnc(CO)c1)=O c1(N(C(CNC(c2c(C)coc2)=O)C)C)nc2ccc([N+](=O)[O-])cc2s1 C(=O)(C1=CC2CCC(C1)C2)N1CC(CNC(=O)C2=C(Cl)CCCC2)CC(C)C1 Cc1onc(C2CCCC2)c1C(=O)NC1CN(C(C2COC2)=O)C2CC12 N1(C(c2c(OC)n[nH]c2)=O)CCCC2CN(C(c3cnc(N)c(Cl)c3)=O)CCC12 c1(OC)cc(Br)c2ccnc(NC(C34CCC(CC3)CO4)C)c2c1 c1(CC)cccc(C)c1C(=O)NCCOCCNC(C1(Br)CC1(C)C)=O c1(CN(C)CC2CCCN2C(C2CC2C2CC2)=O)c(C(F)F)nn(C)c1Cl CC1CCCn2cc(C(=O)NCC3CCC(NC(C4CC(C)(O)C4)=O)CC3)nc21 c1(N(CCC)C)ccc(C(=O)NC(C)CNC(C2CCN(C(=O)OC)C2)=O)cn1 C1(CCC)CN(C(=O)CC(C)(F)F)CC1C(=O)NCC1CCC(=O)NC1 C(c1ccc(F)c(C)c1)=CC(N1CC(NC(Cc2c(C)cc(C)nc2)=O)(CO)C1)=O C1(CNC(C2(C(C)(F)F)CC2)=O)(NC(=O)CCN(C)C)CCC(F)(F)CC1 CC1(C#CC(=O)NCC2CN(C(C3CCCC3)=O)CC23CC3)CC1 CC(C)(C)C(C(=O)N1CCC2(CNC(=O)C2)C1)C(O)C(F)(F)F.c1(SC)nncc(O)n1 N1(CC(=O)NCC(c2cn[nH]c2)=O)CCN(C(=O)Cc2cc[nH]n2)CC1 C1(CC#C)CN(C(=O)CN(C2CCOC2)C(c2ccc(C#C)cc2)=O)CCC1O C1(CN(C)C(c2cc(Cl)cs2)=O)COCCN1C(c1cccc(=O)o1)=O C1(C(=O)OC(C)(C)C)CN(CC(=O)C(C)(C)C)CC12CC2 c1(C(=O)NCC2C(C)CCN(C(CCOCCC)=O)C2)csc2c1CCCC2 C(=O)(CCC(C)(F)F)NC(C1CCN(C(c2nc(C)n(C)c2)=O)C1)C C1(OC)CCC2(C(=O)NC(c3ccccc3)C(=O)NCCCn3nccn3)CC12 c1(C(N2CCCC(NC(COC)=O)C2)=O)[nH]nc2c1COC2(C)C c1(CCCC(=O)NC2(CNC(C(CC)OCC)=O)CCC2)ccccc1Cl c1(C(=O)NC(CNC(C2C(OCC)C2)=O)C)c(C)cc(F)cc1C n1(CCCC(=O)NC2CCC(N(C(=O)COCC(F)(F)F)C)C2)cnc(C#N)n1 N1(C(C=CCOC)=O)CC=CC1(C(=O)NCC(C)OC(F)F)COC C=CC(CC)CC(=O)NC(CO)CCCNC(=O)CCCN1CCCC1 C12(CC(N3CCC(C)(CNC(CN(CCC)C)=O)CC3)=O)CCCCC1C2(F)F N1(C(CNC(CC(C)C)=O)=O)CC=C(C(=O)NC2CCCCC23CC3)C1 N1(CC)CC(C(=O)NCC(CC(C)C)NC(=O)CCc2cc(C)no2)CCC1=O C12(NC(c3ccc(OC)c(Cl)n3)=O)CCCC1N(C(c1ccc(N)cc1)=O)CC2 C(C)(CCCCCO)NC(C(CC)(C)C)c1nnnn1CC(F)F C1(OCC(N2CCN(C(COCCCC#C)=O)CC2)=O)CCCC(C)CC1 O(N(CC)C(=O)C(Cc1cccc(Br)c1)NC(=O)C(C)(O)CC)CC C1(NC(C2(CNC(c3cc(OC)n[nH]3)=O)CCCCC2)=O)CC(C)CC(C)(C)C1 c1(C(=O)NC2CC(OCc3ccc(Br)c(Cl)c3)C2)ccc(C2=COCCC2)cc1F c1(OC)ccc(Cn2nnnc2C2(NCC3CCSCC3)CCC(C)C2)cc1 C1(O)(CNC(c2ncc(N(C)C)cn2)=O)CCN(C(C2(CO)COC2)=O)CC1 N1(C(C2(C(C)C)CCCN2C(C2CSCCO2)=O)=O)CC(C)OCC1C C1(C(=O)NC(CNC(CCN(C)CC)=O)C(C)C(C)C)CCc2ccccc2N1 C1(NC(CCC(C)N(C)C)=O)(CNC(c2ccc(=N)[nH]c2)=O)CCCCC1C Cc1cnc(C(=O)NCCCN2CCN(C(C3CC(O)CN3C)=O)CC2)cn1 N1(C(C(C(C)C)O)=O)CCC(O)C(NC(c2ccc(F)cc2Br)=O)C1 c1(SC)cc(C(=O)NC2COCCC2NC(=O)CCC2CCCOC2)ccc1N c1(N(CCC)Cc2ccccn2)ccc(S(=O)(=O)NCC(C)OC)c(Br)c1 c1(CC)onc(C)c1NCCCN(C(=O)C(c1ccc(Cl)cc1)O)C(=O)N.C(C)C CC(CNC(C1(c2cccc(C(F)(F)F)c2)CC1)=O)C(F)(F)F CC1(CNC(=O)CC2CCN(C(=O)C(O)C(F)(F)F)C2)CCCC1(F)F O=C1NCC2(CCN(C(c3cc(F)ccc3Br)C(=O)NC3COC3)C2)O1 Cc1cc(NC(C2CC2C(=O)NN2CC3(C2)CN(C)C3)=O)ccc1I C1(CNC(COC(C)=O)=O)CCCC(NC(=O)CN(C)CCOC)C1 N12CCC(C1)CCNC(=O)C2C.c1(NCC(=O)NC(C)=O)cn[nH]c1 CC(CCN(C(=O)OC(C)(C)C)C1CC1)C1CC1.C1(=O)C(C)N1CC(F)(F)F c1(C(N(C(C)CCNC(C2CCCS2)=O)C)=O)cnc(O)s1 CC(C)C(CC1CCCC1)C(=O)N1CCC(N2CCN(C(C)CN(C)C)CC2)C1 C1(NC(C2CCC(CC)O2)=O)CCCN(C(=O)CC#N)C1CC c1(C(N(C)CCNC(=O)Cc2cnccc2Cl)=O)cc2n(n1)CCCC2O c1(N(CCCOC)C)ccc(S(=O)(=O)NC(=O)CSCc2nccs2)cc1Cl Cc1c[nH]cc1C(=O)NCc1cc(C(=O)NC(CO)C2(O)CC2)co1 N1(C(CCCC)=O)CCC2CN(C(=O)C(C)(F)C(=O)c3ccccc3)CC2CC1 Cc1nc(C)n(O)c1C(=O)NCC(C)(C)CCNC(=O)CC1CCC(C)(O)CC1 c1(OCC(=O)N(CCNC(c2ccn(CC(C)C)n2)=O)CC)c(C)cccc1C C1(c2cccs2)(C(=O)NCCCCCN(C)C(c2nncs2)=O)CCOCC1 CCC(CC)C(C(=O)N1CCSCC1C(N1CCn2nncc2C1)=O)OC C1(CNC(c2cnc(C)s2)=O)CCCCN(C(C2CC(CCF)C2)=O)C1 C(=O)(CCCCCC(C)C)NC1C(CNC(c2c(C)ccc(OC)c2)=O)CCC1 Cc1ccccc1C(F)(F)C(=O)N1CC(N(C(=O)C)C)C1.C(=O)(C(F)(F)F)N Cn1cnc2ncnc(N(C3CC4(CNC4)C3)C(c3ccc4[nH]ccc4n3)=O)c12 CCCC(CCNC(C1CCN(C(c2cccc3ncnn23)=O)CC1)=O)CCC c1(C(N2CC(CNC(CCC=CC)=O)C3(C2)CC3)=O)sc2ncccc2c1Cl C(=O)(CC(C)CNC(c1ccc(Cl)cc1)c1nnnn1Cc1ccccc1)NC c1(NC(c2cc(C)n(C)n2)c2nnnn2C)ccc(Cl)cc1F N1(c2nc(C)cc(C)n2)CC2CCC(C1)C2NC(=O)Cn1cc([N+](=O)[O-])cn1 c1(C(CCC)(C)O)cn(C2CC(CO)C2)nn1.C12(CC1C(C)C)C(=O)N2 c1(CC)nc(N2CC(C)(C)CC2CNC(C2(C)CCNC(=O)C2)=O)c(F)c(Cl)n1 N1(CC)CCC2(CCCN(C(=O)C(C)(O)C(F)(F)F)C2)C1.c12cccnc1SC2 c1(OC)c(C)cc(C(=O)NCC2(CO)CCN(C(=O)OC(C)(C)C)C2)cc1Br c1(C(=O)NC(C)C(=O)NCC(C)CNC(=O)CC2CCOCC2)nocc1Cl CC1CN(C(=O)CCC2(C)CC2)CC(C(=O)NC2CC(CCF)C2)O1 c1(CC(=O)NC(C2CCCC2)CNC(CCC(C)OC)=O)ccc2occc2c1 C1(C(=O)OCC)CCN(C(c2ncn(C)n2)=O)CC1C c1(C(=O)OC(C(CNC(C(CCOC)OC)=O)(F)F)=O)ccc(F)c(C)c1O CC(C)C(CO)N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC3(C)CCCCO3)cc2s1 N1(CC)CC2CN(C(C3CC(O)CN3C(=O)CCC(=O)NC)=O)CC2C1 C(=O)(CCS(N)(=O)=O)NC1CC(CNC(C(c2c(OC)cccc2)=O)=O)C1 N1(C(c2n(C)nc(Br)n2)C(=O)NCCCF)CCC2(COC(C)(C)C2)C1 C1(C(F)(F)F)(C(=O)NCCNC(=O)C=CC(=O)NC2CC2)CC2CCC1CC2 C1CCCC(=O)N1.N1(C(C2CCC(CNC(N)=O)O2)=O)CCOCC1C1CC1 C1(NC(C2(CC)CC2)=O)CC2CN(C(c3coc4c3CSC4)=O)CCN2C1=O Cc1noc(-c2cn(CC(=O)NCC(C)NC(=O)CCCn3cccc3)cn2)n1 CCS(=O)(=O)CC(=O)NC1CC1CNC(C1CN(C(C)C)C1)=O c1(C(=O)NCC(CNC(C2(CC)CCC2)=O)(C)O)ccccc1C1CC1 N1(C(C(=O)N(C(c2ncc(C(F)(F)F)s2)C)C)=O)CC(O)CC1C(=O)O c1(C(N2CC(CC=C)(C(N3CC(N(CC)CC)C3)=O)C2)=O)ncncc1N C1(OC)CCN(C(=O)C(CNC(=O)C(C)C2CCCC2)N(C)C)CC1(C)C C1(N(C(=O)CCSCC(N)=O)C)CCN(C(c2ccnn2CC(F)(F)F)=O)C1 c1(C(=O)NC(C2CCN(C(c3ccc(C4CC4)o3)=O)C2)C)nsc2ccccc12 N1(C(c2c(C)[nH]c(C)c2C)=O)C2COCC1CN(C(=O)CC(F)(F)F)C2 CC(CC(F)F)C(=O)N(C1(CC(N2CC(O)(C3CC3)C2)=O)CC1)C C1(C(=O)NC2CCC(OC)C2)CC(C)CN(C(c2ccsc2)=O)C1 C1(NC(CCC(C)N(C)C)=O)CC2CC(NC(C3CC(O)C3)=O)C1C2 C1(CNC(C(CC)OC)=O)CN(C(c2ccc(C(C)=O)cn2)=O)CCC1(F)F N1(Cc2c(OC)c(Cl)ncc2)CCC(P(C)(C)=O)C1 c1(CSc2nc(C(C)OC)nn2-c2ccc(Cl)cc2)c(C)nc2ccccn12 C#CC1CN(C(c2[nH]cc3c2CCCC3)=O)CCN1C(=O)C=C1CCOCC1 Cc1cnc(F)cc1-c1nc(C(=O)Nc2ccc(Br)nc2O)cs1 C(=O)(C(C(C)C)C(C)C)NCc1occ(C(=O)NC(C(C)SC)C)n1 Cc1ccc(F)c(C(=O)NC(CCF)C(=O)NCCCC2CC2)c1 c1(C(=O)NCC(CC)NC(c2ncnn2C)=O)ccc(S(C)(=O)=O)[nH]1 C(=O)(C1CCc2cccnc21)N(CCCN(C(c1c(OC)cccn1)=O)C)C Cc1cc(C)c(C#N)c(CCCNC(=O)CC(C)SC2CCCC2)n1 CCCCCCCCC(=O)N1CCCC1CNC(c1cnn(C2CC2(F)F)c1)=O C1(C(=O)NC(c2ncc[nH]2)C)CC12CCN(C(=O)CSC(F)(F)F)C2 N#Cc1ccc(C(N2CCC(CNS(=O)(=O)CCl)C(O)C2)=O)cc1.C(CC=O)N N1(C(CCSC)=O)CC2(CNC(c3cn(C)nc3-c3ccoc3)=O)CC1CO2 N1(C(c2ccc(N)c(N)n2)=O)CCCC2(CNC(=O)C3=NOCC3)CCCCC12 C12(C(=O)NCC=CCNC(C(Cc3ccccc3)OC)=O)CCC(C)(CC1)CC2 C(=O)(C#CC1(CC)CC1)N(CCC)CCNC(=O)CC1OCCC1C Cc1nn(C)c(Cl)c1C(N1CC(NC(=O)CNC(c2ccccn2)=O)C(C)C1)=O N1(C(c2c(C)nc(C)o2)=O)CCC(NC(C2CCCSC2)=O)CC1C c1(C2COCC(C)O2)ccc(Nc2nccnc2C#N)cc1F C1(C(=O)NC(C)CCCCCO)CN(C(c2cn(CCO)nn2)=O)C2(CCC2)C1 C1(F)(CNC(C2CC2(F)F)=O)CCCN(C(=O)Cc2cnccn2)CC1 N1(C(C(CC=C)(F)F)=O)CCCCC(CNC(=O)C(c2cnn(C)c2)O)CC1 C1(C(N2CCN(C(CC(CC)(C)C)=O)C(C3CCC3)C2)=O)CCc2n[nH]cc2C1 CCCC(C(=O)NCCCN(C(=O)CC1NC(=O)NC1=O)CC)N(C)C CC1CCC(OCC(=O)NC2CCCCC2N(C)C)CC1 c1(OCC#C)cccc(C(=O)NCC2(CNC(C3COCCO3)=O)CC2)c1 CC(O)C(C)C(=O)N(C1CCCC1)CCNC(=O)CNC(=O)CCC1CC1 C(=O)(CCC(=O)NC(C)CN(C(=O)C(n1ccc(C)n1)C)C)NCC N1(C(CSCC=C)=O)CCCN(C(=O)CC2CCOCC2)CC1C N1(C(C(C)C2CCCCC2)C(=O)NCC(F)F)CCS(=O)(=O)C2CCCC12 CC(C)C(C)C(C)CC(=O)N(C1CCN(C(c2ccn3c2CSCC3)=O)CC1)C C1(NC(C=Cc2cn(C)nc2)=O)CCN(C2CCN(C3CC3)C2=O)CC1F Cc1ncccc1CC(=O)NCc1cc(C(=O)N(C)CCc2ccccc2)on1 CC1=NN(C)C(=O)C1CC(N1CCC(N2OCC(C(=O)OC(F)F)C2=O)CC1)=O c1(C(=O)NCC(CNC(C(=Cc2cnc[nH]2)C)=O)C)cc(Br)n(C)n1 C(=O)(CS(=O)(=O)c1ccccc1C)NCC1CCN(C(C(C)=C(C)C)=O)C1(C)C Cc1nc(NCCCc2ccncc2)cc(NC2CCOCC2C#N)n1 Cc1cc(C(N2CCCC(O)(CN(C)C(C3(C)CCCS3)=O)C2)=O)cc(N)c1O C(C(CNC(C1C2CC(=O)CC12)=O)S(C)(=O)=O)NC(C1(CC)CCCCC1)=O C1(NC(C(C)N(CC)CC)=O)C=CCN(C(=O)CCc2cnoc2)C1 C(=O)(C(C)(C)S(C)(=O)=O)N1C(C2(NC(C3CCC(CC)O3)=O)CC2)CCC1 Cc1cccc(C2(C(N3CCC(F)(CNC(c4cccc(O)n4)=O)C3)=O)CC2)c1 N1(C(=O)NCCC(c2ccc(C(C)(C)C)cc2)(C)C)CC2C=CCOC2C1 C(CCCCCNC(=O)CCN1C(=O)CNC1=O)N(C(C1C(CC)OCC1)=O)C C(c1cccc(Cl)c1)=CC(=O)NCC1C2CN(C(c3ccn(CC)c3C)=O)CC21 Cc1ccc(F)cc1CC(N1CCC(C2CCCN2C(C23CC(C)(C2)C3)=O)C1)=O c1(C(=O)NCCC(CC)(CC)NC(=O)CC(C)COC)cn(C)c(=O)nc1O C1(C#N)(C(N2CCC(NC(CSC(C)(C)C)=O)C2)=O)CC(=O)C1 C#CC1CN(C(=O)Cc2cncs2)CCN1C(=O)C1=COCCC1 N1(C(C(C)(C)OC)=O)C2COCC1CC(NC(C1CC1c1cccnc1)=O)C2 C(=O)(CCCCCF)NCCNC(CCCNC1CCN(S(C)(=O)=O)C1)=O N1(C(C2=NOC(C)C2)=O)CCC(CNC(c2ncccc2N(C)C)=O)C(F)(F)C1 Cc1scc(C(=O)NC2(CO)CCN(C(=O)C(c3ccc(Cl)cc3)(C)O)C2)c1N C1(NC(CC2(C)CC2)=O)CN(C(c2cc(=O)c(Br)c[nH]2)=O)CC2(CC2)C1 c1(C(N2CC(OC)C(NC(C3C=CCC3)=O)C2)=O)cccc2[nH]c(=N)oc12 c1(OC)cc(CC(=O)N(C2CN(C(=O)Cc3ccon3)CCC2C)C)ccc1Cl C1(C(=O)OC)Cc2ccoc2CN1C(c1cnn2c1CCC2)=O O=S(=O)(C=Cc1ccccc1)N1CC2CN(Cc3ccc(O)cc3Br)C2C1 c1(C(=O)NCC(CC)NC(=O)CCOCC(F)F)c[nH]nc1COC N1(C(C2(C)CN(C(C3CC3(C)C)=O)C2)=O)CCC2(CNC(=O)N2)C1 C1(NC(c2c(C(C)C)n(C)nc2)=O)CCC(C)N(C(C2C3CCCCC23)=O)C1 CC1CN(C(c2cnn(CCF)c2)=O)CC(CCNC(C2(O)CCC2)=O)O1 c1(C(=O)NCCC(C)CCNC(=O)C2=CCCCO2)cc(Br)c(C#N)s1 C1(NC(CCC#C)=O)CCN(C(=O)CCCC(=O)NCCCC)CC1F C12(C(=O)NCCC3N(C(C4CC(F)(F)C4)=O)CCCC3)CCC(O)(CC1)CC2 Cc1ccc(O)c(C(N2CCCC(NC(=O)C=CC3CCOC3)C2)=O)n1 C=CCCC(C)(C)C(=O)NCC12CC1CN(C(c1ncc[nH]c1=O)=O)C2 c1(C(C)C)onc(C(F)(F)F)c1C(=O)NCC(O)CNC(C12CC(C)C1C2)=O c1(C(N2CCC(C)C2CNC(c2cnc(C(N)=O)s2)=O)=O)cc(F)ccc1Cl c1(C(=O)NCC(C)N(C(=O)CN(CC)CC2CC2)CCC)ccccc1C c1(OCC(=O)NCC(CNC(c2ncc(C(F)F)s2)=O)CO)cccnc1Cl CN1CCC(NC(=O)CCCCCCNC(C2COCCO2)=O)C(C#N)C1 N1(CC(=O)NCCC(=C)CNC(=O)CS(=O)(=O)N(C)C)CCc2ccccc2C1 C1(C(C)NC(C(C)NC(CC)(C)C)=O)CCN(C(c2nnn(C)c2N)=O)CC1 C1(F)(C(=O)NCC(CCCC)NC(=O)CSS(C)(=O)=O)CC2(CCC2)C1 C1(CNC(Cc2cccc(CC)n2)=O)CN(c2ncc(CC)cn2)CCC1(F)F C#CCC(C(=O)NC(CCSC)C(=O)Nc1cnn(CC)c1C)C1CC1 Cc1cc(C(=O)NCC2CC2NC(C2CC3CCC(C2)O3)=O)cnc1O C1(C(=O)NCC(C2CCCCC2)NC(=O)C=CCO)CCNC(=O)C1 C1(NC(C=C(COC)C)=O)COC2(CCN(C(C3(F)CCC3)=O)CC2)C1 C1(C(N2CCN(CC(C)C)CC2)=O)CN(C(c2cncc(O)c2)=O)CCC1(F)F c1(C(=O)NCC2N(C(C3(C)CC3)=O)CC2)cnc(N)c(-c2ccccc2)c1 C(=O)(C(O)C(F)(F)F)NCc1cn(CC(C)NC(Cc2cnc(C)s2)=O)nn1 C1(C(=O)NC2CCC(CN=c3[nH]nc(C(C)(C)C)o3)C2)Cc2ccccc2O1 N1(C(C(C)OC(C)C)=O)CC2(CC(NC(=O)Cc3csc4nccn34)CO2)C1 N12CC3ON=C(CN1C)C3C2.c1(CC2(C=O)CC2)cccnc1.C1(C)(C(=O)N)CC1 CC(C)C(C(=O)NCC1CC(C)CN(C(=O)CCOCCN(C)C)C1)C(C)C c1(C(=O)NC2CCC(NC(CC(=O)NCC)=O)C2)cc(Cl)c(Cl)cc1N N1(C(C2N(C(c3cc(C)n(C)c3)=O)CCN(C)C2)=O)CC2(CCC(=O)NC2)C1 N1(C(CC(CNC(c2c(OC)cncc2)=O)O)=O)CCC(F)(F)CC1 C(=O)(C#CC1CCCC1)NC1C2CN(C(Cc3cccc(C#N)c3)=O)C1C2 CCCC(C)C(=O)N1CCOC(C(=O)NCc2[nH]c(C)nc2C)C1 C(=O)(C(CC(C)C)ONC(=O)C(F)CC1CCOC1)NCCSCCC=C C1(C(=O)NC2C3CC(NC(C4N(CC)CCCC4)=O)CC32)COC2(CCC2)C1 C(=O)(C1=Cc2cc(F)ccc2OC1)NCC1C2CN(C(C=C(CCC)C)=O)C1C2 c1(C(=O)NC23C(CN(C(C4(CC)CC4)=O)C2)C3)ccccc1[N+](=O)[O-] Cc1ccc(C(=O)NC(C)C(CO)NC(c2ccc(C#N)o2)=O)cc1C(C)(C)C N1(C(C=CC(C)NC(c2ncc(F)cc2N)=O)=O)CC(P(C)(C)=O)C1 C1(NC(CC2(COC)CC2)=O)C2CCC1CC(NC(=O)C(C)CC(N)=O)C2 c1(C(=O)N(C(c2ccccc2Cl)CCC)CC=C)ccc(OCC)cc1 CCCC(C)C(=O)N1CCCCC1CN(C(=O)CNC(N1CCCC1)=O)CC C(=O)(C(=O)C(C)CC)NC(C(=O)NC(CC)CC)CCF CCCCCC(O)C(=O)NCC1CCC(CNC(c2cc(N)cc(F)c2)=O)CC1 C123CC(CO1)N(C2)C3.CS(C)(=O)=NCCNC(C1CCN(C(N)=O)CC1)=O C(=O)(CC1CCCc2ccccc21)NC(CC)CNC(c1nc(=N)cc[nH]1)=O C(=O)(C1=CCCSC1)NC12CC(NC(c3n(CC#C)ccc3)=O)(C1)C2 CC1(C)CCC2CCN(C(c3ccc(-c4coc(O)n4)cc3)=O)C=CC=C12 Cc1c(OCC(N2CCN(C(C3CC3(C)C)=O)C(CCO)C2)=O)cccc1Cl N1(C(COC(C)(C)C)=O)CC(NC(=O)CC2CC2C2CC2)C(C2CC2)C1 Cc1cnc(C(=O)NCC(C)(C)CNC(=O)C(C)OCC(C)C)c(Br)c1 C(c1ccc(C(=O)O)o1)=CC(=O)NCCc1nn(CC#C)c(=O)o1 c1(OCC(=O)NC2C(NC(=O)CC3CC=CC3)CC2)cccc(C(F)(F)F)c1 c1(C(=O)NCCC2CCN(C(C(CC)(C)C)=O)C2)ccc(C#N)c(C)n1 c1(C(N(CC(CNC(c2scc(C)c2C)=O)O)C)=O)cc2ccccn2n1 C1(NC(C2CCCC(=O)N2)=O)CN(C(c2cnn(CCO)c2)=O)C2(CCOC2)C1 C1(C(=O)NCCN2CC(OC)C2)CCN(C(=O)C#CC(C)(C)O)C(C)(C)C1 c1(NC(CCc2cn(-c3cccc(OC)c3)nn2)=O)c(Cl)ncc(Br)c1C N#Cc1ccc2c(=NC(=O)N3CC=C(Cc4ccccc4)CC3)[nH][nH]c2c1 C1(C(N(CCSCC(=O)NCCOC)C)=O)CCOC1c1nccn1C C12CCN(CC1)C(=O)CC2.C1(C)CCN1C(=O)C(C)=C1CC1.C#CCC c1(N2C(CNC(c3nccc(CC)c3)=O)CC2)ccn2c(Br)cnc2n1 CC1CN(C(C2CCCO2)=O)CC1NC(=O)C=CCOc1ccccc1 N1(C(CC(CC)NC(=O)Cc2cccnc2)=O)CCC12CCOCC2 C1(C(N(CCNC(C(C2CCCC2)OC)=O)C)=O)CCCCCC1(F)F N1(C(C(CCC)OC)=O)CC2CCCC(CNC(C3CCOC3)=O)C2C1 N1(C(c2cccc(F)c2F)=O)C2CCC1CN(CCc1cc(Cl)ccc1Cl)CC2 C12(CNC(C3=NOC(C)C3)=O)CCCC1CCN2C(c1cnn(C(C)(C)C)c1)=O c1(C(=O)NCC(C)(C(C)C)NC(C=CSC)=O)ccnc2c1cnn2C CCN=c1[nH]c(C)c(C(=O)NC2(CNC(C3CC(C)(C)OC3=O)=O)CC2)s1 c1(C(=O)NC(C2CCN(C(c3nc(CC)sc3)=O)C2)(C)C)ccc(N(C)C)cc1 c1(NC(C2C3CN(C(c4c(CCC)[nH]cc4)=O)CC32)=O)ccc(F)cc1C c1(C(=O)NCC2CC(NC(Cn3nnc(C)n3)=O)C2)c(C)nn(C)c1Br C(=O)(C1CCCc2nnn(C)c21)NC(C)CNC(c1ccc2oc(O)nc2c1)=O C(=O)(C1CCc2cccnc21)N1CCC(O)(CNC(CCOCC#C)=O)C1 N1(C(=O)C=Cc2ccoc2)CC2CC2(C(=O)Nc2csnc2C2CC2)C1 c1(OC)ccc2nc(C)cc(C(=O)NCC(CC(=O)O)c3ccc(F)cc3)c2c1 C1(CC#C)(C(=O)NC2CCC2CNC(C2CC=CCC2)=O)CCCCC1 C1(C2CCN(C(=O)CCCc3csc(=N)[nH]3)C2)(NC(CC=C(C)C)=O)CC1 C1(C(=O)NC2CCC(NC(c3cc(C)c(C)o3)=O)CC2)CCC(C2CC2)C1 C1(C)C(=O)NN2CCCC2CN1C(c1ccoc1)=O.CCS.CC C1(CNC(c2coc(C3CC3)n2)=O)COCCN(C(=O)CCc2cncnc2)C1 CC1OCCN(C(=O)CCS(C)(=O)=O)C1C(=O)Nc1ccc(O)cc1C1CC1 CCC(CC)C(C)C(=O)NCC(c1ccc(F)cc1)NC(c1snc(Cl)c1Cl)=O C(=O)(N=c1ccn(CC2CC2)[nH]1)C1C(NC(CCCCSC)=O)CCCCC1 C(=O)(NNC(=O)OCC)NCC=C.C12(CC1C(=O)OC(C)(C)C)C(=O)OC2.C(C)(C)N N1(C(C2(C#C)CCCCC2)=O)CC2C=CC1C(C(=O)NCCCCCC)C2 C1(C(=O)Nc2c(SC)nccc2)CC2(CCN(C(=O)C(C)(F)F)CC2)CO1 C1(CNC(c2cc(C)sc2)=O)CN(C(c2cc(C(N)=O)n(C)n2)=O)CCC1C N1(Cc2c(OC)nc(Cl)cc2)C2CCC1CN(c1ccnc(N3CCCC3)n1)C2 Cc1oc2nc1C(=O)N(CCCO)C2.c1(OCC(=O)NCCCO)cccnc1 C(c1cnccc1C)=CC(=O)NC1C(CNC(CC(COC)C)=O)C1 c1(C2(C(=O)NC(CNC(Cc3c(C)occ3)=O)CO)CC2)cccc(F)c1 Cc1ncnc(O)c1C(N1CC(NC(C2(CF)CC2)=O)CC(O)C1)=O c1(C(C(=O)N(CC(C)CNC(=O)CC2COCCO2)C)(C)O)ccc(F)cc1 Cc1noc(C)c1C(C)CC(=O)NCCOCCNC(=O)Cc1cccn1C Cc1ccc2c(C(=O)NC3CC(CNC(C4CCCCC4)=O)C3)ccnc2c1 C1(C(N(CCSC)CC)=O)COC2(C1)CN(C(=O)C=C1CCC1)C2 CCN(OC)C(=O)CN=c1[nH]c2cc(Cl)c(S(=O)(=O)NC(C)(C)C(C)O)cc2s1 c1(C(N(C2CCCC(NC(c3nn(C)cc3Cl)=O)C2)C)=O)cn2c(n1)COCC2 c1(C(=O)NCCN(C(=O)CC23CCCC2C3)CC)ccc(Cl)c(-n2nnnc2C)c1 c1(C(C)=O)ccc(C(=O)NCC2CC(F)CN2C(=O)C(C)=C2CCC2)nc1 c1(C(=O)NC(CC)CN(C)C(C2CC(OC)C2)=O)c(C)sc(C)c1C#N C1(CSC)CCN(C(=O)NCCN(C)Cc2cccc(-c3ccccc3)n2)CC1 C1(C(N2C(C)(CC(=O)NCC#CC(C)C)CC2)=O)CCCN(C)C1 N1(C(CCCCSC)=O)CC2CCCC(NC(c3cncc4c[nH]nc34)=O)C2C1 C1(CNC(=O)CC(F)F)CN(C(=O)CN2CCCCCC2)C2CCN1C2 C1(C(=O)NC(CCOC)(C)C(=O)O)CC(=O)OC12CCCCC2 S(=O)(=O)(C1CC1)NCC(N1CC(CNC(CO)CCc2ccccc2)C1)=O c1(C(=O)NCCCN(C(C2CCCC(C)C2)=O)C)csc2ncnc(O)c12 CN1CCN(CCC(N2CCC(CNC(=O)C3=CCSC3)CC2)=O)CC1 c1(NCC(C)C)cc(Cl)ccc1C(=O)NCC1CC1NC(c1c(O)noc1C)=O c1(NC(C(c2c(C)n(CC(C)C)nc2)N2CCC3CC3C2)=O)cccc(Cl)c1C N1(C(c2cc(COC)oc2C)=O)CC2CCN(C(c3nccnc3C)=O)CC2C1 c1(C(=O)OC)cc(C(=O)NCCCC(C)NC(=O)CC2CC(C)C2)ccn1 C12(C(=O)NC(C3CCCC3)C#C)CCCC1CN(C(C1CCC(C3CC3)C1)=O)C2 N1(C(C2COCCOC2)=O)CCC(C2(O)CN(C(=O)CC3CCOC3)C2)CC1 c12cc(cc(C)c1)C(=O)N1CCCCC1C(=O)N2.C1(NC(=O)OC)CC1OC C(C(C)CNC(=O)CC1C=CCC1)NC(C1(CC(C)C)CC1)=O N1(C(CSCCC)=O)CC(CNC(c2ccc(NC(=O)NC)cc2)=O)CC1(C)C N1(C(=O)OC(C)(C)C)CC2(CC1C(=O)NCCCCO)CC(F)(F)C2 C1(NC(C=CC(=O)OCC)=O)CCOCC1NC(C1CC2CC2C1)=O c1(C(N2CCCC(F)(CNC(c3ccnc(C)n3)=O)C2)=O)cc(F)c(F)cc1O c1(NC(c2c[nH]nc2-c2ccc(Cl)cc2)=O)ccc(-c2ccc(F)cc2)cc1F c1(C(=O)NC(C)(C)C)ccccc1C(N1CC(N(C)C(c2cnsn2)=O)C1)=O c1(C(=O)NC2C3CN(C(C(C4CCC4)OC)=O)CC32)cc2n(n1)CCCC2 C1(C(=O)NCC2(O)CC(NC(c3cncc(Cl)c3)=O)C2)C2(CCC2)C12CCC2 c1(CC)ccc(NC(c2coc(C(C)OC)n2)=O)cc1.C1(=O)CC=CCN1 N1(C(C2(N(C)C)CCOCC2)=O)CCCCC(NC(C2(C)CCCNC2=O)=O)C1 NS(=O)(=O)c1ccc(COC(=O)Cn2ccc(=O)n(C(=O)c3cscn3)c2=O)o1 N1(CC(=O)Nc2c(Cl)ccc(OC(CCC)C)c2)C(=O)NC(C)(C2CC2)C1=O Cc1noc(C)c1C=CC(=O)NC1(C)CCCC1NC(c1c[n+]([O-])c(C)cn1)=O N1(C(C(CNC(c2cnnn2C)=O)OC)=O)CCCC(O)(CO)C1 Cc1noc(C(=O)NCC(O)CNC(C2CC2C2CCC2)=O)c1C(F)(F)F C1(c2nc(C(C)C)[nH]n2)CCCCN1C(c1ccnc(OCC2CC2)c1)=O S(=O)(=O)(c1cc(C(=O)NC(CNC(C2(S(N)(=O)=O)CCC2)=O)C2CC2)co1)NC C1(NC(C(C2CC2)NC(C2CC3(CCC3O)C2)=O)=O)C2CCC(C2)C1CO c1(CN(C(c2cn(C)nc2Br)C(=O)NC(CC)C)C)cc(Cl)ccc1F c1(C(=O)NC(=O)C(N2CC(COC)CCC2=O)=O)ccc([N+](=O)[O-])s1 C1(C)(NC(C2(CNC(C(C)OCCOC)=O)CCCO2)=O)CCCC1(C)C C12(C(=O)NC(C)(C)CCNC(=O)CC3CCC3)CC1CNC2=O N1(C(Cc2cccc(OC)c2)=O)CCC2CCCC12C(=O)NCCN1CCCCC1 c1(C(N2C3C(NC(CCOCC(C)C)=O)C(C3)C2)=O)ccc2c(n1)CCOC2 c1(C(C(=O)NCCCN(C)C(C2C3CC4C(C3)C24)=O)C2CC2)ccc(F)cc1 N1(CC)CCCC(N2CC(O)C2)C1.c12nc(co1)CC(=O)NC(=O)CO2 N1(C(C2(OC)CCOC2)=O)CCC2(C1)CN(C(c1ccn(C3CCCC3)n1)=O)C2 c1(C2(C(CCC)=O)CCC2)cc(C)no1.C1(=O)CSCC2C(C2)C(=O)N(C(C)C)O1 Cc1conc1CC(=O)NC1CC(O)C1CC(=O)NC(c1nnc(C)o1)C CC(O)C(F)(F)C(=O)N1CC(NC(c2sccc2-n2ccnn2)=O)C1 C12(NC(C3C(C(=O)OC)CC3)=O)CCOCC1CN(C(C1(C(N)=O)CC1)=O)C2 Cc1cc2c(C(=O)NC3(C)CN(C(c4c(Cl)n[nH]c4C)=O)C3)cccc2o1 C(=O)(C(CNC(C1(C)CC(C)(C)C1)=O)CC(C)C)Nc1c(C)nn(C)c1 C1(CN(C)CC)CCN(C(c2ncoc2CNC(C2CC23CC3)=O)=O)C1 N1(C(c2ccn(C)c2)=O)CCC2(CC1)CC(NC(c1c(Cl)ccnc1Cl)=O)C2 C(C)(CC(=O)NC(C1(CNC(c2cc(CC)no2)=O)CC1)C)=CC C1(NC(c2cc(CNC(c3c(CC)onc3C)=O)ncc2)=O)CCCCCC1F CC(C)C(F)(CNC(=O)CCCN(CC(C)(C)C)C)C(=O)NOCC1(C)CC1 n1(CC)nc(C)c(C(=O)NCC(CC(F)(F)F)NC(C2CCCCO2)=O)c1Cl CC1(C(=O)NC2CC(C(=O)Nc3cccc(CO)c3)C2)CCCOC1 N1(C(c2cncc(OC)n2)=O)CCn2ncc(CN(C(=O)C(C)SC)C)c2C1 c1(SCCOCC(N2CC(C)(OC)C2)=O)ccccc1Cl C(=O)(C#CC1CCOC1)NCc1ccc(C(N(C)Cc2cnnn2C)=O)cn1 N1(C(c2c(Cl)ccc(OC)c2)=O)C2CC(F)C(C2)C1C(=O)NCc1ccc[nH]1 N1(C(CC(C)C(F)F)=O)CCC(NC(=O)C(F)(F)c2nccn2C)CC(O)C1 C1(C(=O)N(C)Cc2ccns2)(COC)C=CCN1C(=O)Cc1nocc1C N1(C(C(C)NC(C)=O)=O)CC(NC(C23CCCC2C3(F)F)=O)CC12CCOCC2 C(c1ccccc1Cl)=C(C)C(N1CCN(C(c2c[nH]c(C#N)c2)=O)C(C)C1)=O CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NCC(C)(CO)NC(C12COCC1C2)=O CC(C)CS(=O)(=O)CC(=O)NCC1CC(CNC(C2C=CCC2)=O)C1 N1(C(=O)Nc2ccc(CC)cc2)CC2CCC(C1)C2NC(=O)C1CC1 CC1CC(CNC(=O)C(c2cnn(C)c2)O)CCN1C(=O)CC1CCCCC1 CCC(C(=O)N1CC(N(C(=O)CN(C)CC)C(c2cccs2)C)C1)SC Cc1cc(C#N)cc(C)c1NC(C1CCN(C(c2cccnn2)=O)CC1)=O C(CC(CNC(C1(C(C)(F)F)CCC1)=O)NC(C1CCOC1)=O)OC C12(CNC(c3cc(CC)on3)=O)CCCCC1N(C(=O)C(C)C1CCOC1)CC2 CC(F)(C(=O)NC1CCCN(c2nccnc2Cl)C1)C(F)(F)F CN1CCN(C(=O)CN2CC3CC3C2)C(CNC(=O)C(F)F)C1 N1(C(Cn2c(C)cc(C)n2)=O)C2CCC1CC(NC(C1CC3CCC(C1)C3)=O)C2 S(=O)(=O)(c1cccc(Cl)c1)N(CCNC(c1c(C#N)ccnn1)=O)CC1CC1 N1(C(c2cn(CC)nc2C)=O)CC2CC1CN2C(=O)CCCN1CCOC1=O c1(OCC)ccccc1N1CCC(C(=O)NCC2NCN(C)C(=O)C2N)CC1 c1(OCCC(=O)NCC2(O)CN(C(C3CSCCS3)=O)C2)ccccc1 C1(CNC(c2cccc(F)c2)CC)CCC2(CCCCCC2)O1 c1(C(N2C3CC(NC(COC(CC)C)=O)C(C3)C2)=O)cnc2ccccc2n1 Cc1csc(CC(=O)NC2CC(CCC(=O)NCC3(N(C)C)CC3)C2)n1 c1(C(=O)NC2CC(CCNC(C(C)n3cccc3)=O)C2)cc2cn[nH]c2cn1 N(C(=NCC(C)C1(C)OCCO1)NCC(C)C)CC1CCN(C(C)=O)C1 N#CCC(CCc1ccccc1)c1ccccc1.N1(CC(=O)N)CCCCC1=O N1(C(C(CC#C)C)=O)CC2CCC2(CCNC(=O)C=CCN(C)CC)C1 c1(C(=O)NCCNC(=O)COC2CCOCC2)ccc2c(O)nccc2n1 N1(C(C(C)N2CCC2)=O)CC(O)(C(F)C(=O)NC2CC=CC2)C1 C1(C(=O)NCCCNC(Cn2cc(C(=O)OCC)nn2)=O)CC(C)C1(C)C Cc1cccc2c(C(N3CC4CCN(C(=O)C(C)CC5CC5)C4C3)=O)csc12 N1(C(C=CCCC)=O)CCN(C2CCC(NC(=O)Cc3cc[nH]n3)C2)CC1 N1(C(CC2(CSC)CC2)=O)CCCC2(CCN(C(=O)C(C(C)O)N(C)C)C2)C1 C1(C(=O)OC)CC(=O)N(C)C1C(=O)NCC1CN(C(C2CCC3(CC2)CC3)=O)C1 C1(C(=O)NCC(C)(O)C2CCC2)CSCN1C(C1CCCCO1)=O N1(C(c2occ(C)c2C)=O)CC2CCC1CN2C(c1csc(C(C)(C)C)n1)=O n1(CC)nc(C)c(C(=O)NCC2(O)CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)c1Cl N1(C(CCCSC)=O)CCC(F)C(NC(c2ccc(C(=O)OC(C)(C)C)cc2)=O)C1 c1(C(C)Nc2cc(Cl)ncc2Br)ccc2c(c1)OCCO2 C1(C(N(CCNC(CSCC=C)=O)CCOC)=O)CCCOC1c1ccccc1 c1(C(=O)NC(CC)CNC(c2cc(O)n(C)n2)=O)nccn2c(Br)cnc12 c1(C(C)C)cccc(C(=O)NC2(CNC(c3ccc(Cl)s3)=O)CCOC2)c1F CC1CC(=O)NC1C(=O)N(CCCCN(C)C(C1(C(F)F)CCOCC1)=O)C Cc1c(O)ccc(C(N2CC3(C2)CN(C(=O)CN(C)C(N)=O)C3)=O)c1C C1(NC(C2C(C)(C)CC2)=O)CCCCCN(C(=O)C=CCOC2CCOCC2)C1 C(C1CN(C(C2CCSC2)=O)Cc2ccccc21)NC(c1nn(CC)c(C)c1)=O Cc1ccc2c(c1)CCC(C(=O)NCCCNC(=O)Cc1c[nH]nc1C(F)F)O2 CCC(C)C(C(=O)NCC(O)CC(F)(F)F)NC(=O)CCNC(=O)CO CCC(F)(F)C(=O)NC1CCCC(CNC(C2(S(N)(=O)=O)CC2)=O)C1 N1(C(CCS(C)=O)=O)C2COCC1CC(NC(C1CCCN1C(N)=O)=O)C2 S(=O)(=O)(c1ccc(C)c(C)c1)NCCC(=O)OCCc1c(OC)ccc(Cl)c1 c1(C=O)ccnc2cc[nH]c12.C(C)(CCCc1ccccc1)NCCN(CC)CC Cc1ccccc1C=CC(N1C(C(=O)NCCOCCOC)CCC1C1CC1)=O C(=O)(C(CNC(C1(C)CNC(=O)C1)=O)C(C)(C)C)NCc1c(C)cc(C)s1 Cn1cc(NC(C2CCN2C(=O)C(c2ccc(F)cc2)=O)=O)c(C(N)=O)n1 CCCC(C(O)C(=O)NC1CC(C2CCC2)C1)NC(C1CN(C)C1)=O N1(CC)CCOCC1C(=O)NCC1CCOCC1C(N1CCCC1)=O.C1CON1 C1(S(C)(=O)=O)(C(=O)NC2C(NC(C3(N(C)C)CC3)=O)CCC2)CC(O)C1 c1(NC(c2cc(NC(COCC)=O)cn2C)=O)cccc2nc(CC)[nH]c12 N1(C(C2(CC)CC2)=O)CCC2CC(C(N3CCC(F)(F)CC3)=O)C2C1 C(=O)(CC(C)(C)CCC)NCC1(CNC(C2(C=C)CC2)=O)CC2CCCC2C1 c1(C(=O)NC(CC)CNC(=O)CC2(OC)CC2)cccc(-c2nnco2)c1 C=CCC(CNC(=O)C(CC)CC)C(=O)N(C)C(C1CCCC1)C C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCN(c1cc(Cl)nc(C(F)F)n1)C)C C1(CC(=O)NC(C)C)(OCC)CN(C(=O)C(C)COC(C)COC)C1 CC1CCCN(C(C2(O)CC(CF)C2)=O)C1CCNC(c1cccc(CF)c1)=O Cc1nn(CC(=O)NCC(C)NC(=O)CSc2ccncc2)c(C)c1Cl N1(C(C2C(=C)CC2)=O)CC(C(F)(F)F)CC1CNC(=O)CCc1nc(CC)no1 N1(C(C(c2ccn(C)n2)C)=O)CCC2CCN(C(=O)CCc3cnco3)C2C1 C1(NC(C2CCC(NC(C(C)C3CC3)=O)CC2)=O)CCC2(CCCC2)C1 C1(NC(C(C(CC)C)OC)=O)C(C)CCN(C(C2CN(C)C(=O)N2)=O)C1C c1(C(=O)NCC(CNC(Cc2c(C)cco2)=O)(C)O)csc2c1CCCC2 c1(C(CC)NC(Cn2cc(C3(N(C)CC)CCC3)nn2)=O)cccc(Cl)c1 c1(C(=O)NC2CC(CNC(c3nc(CC)oc3)=O)C2)ccc(OC(F)(F)F)cc1 Cc1cc(OCCCN(C(C2CCc3cnn(C)c3C2)=O)CC)ccc1[N+](=O)[O-] Brc1ccc2[nH]cc(CN3CCC(OCC4CCCO4)CC3)c2c1 c1(C(=O)NC2CN(C(CCCOCC)=O)C2)n[nH]c(CC)c1Br C=CC(C)(CC)NC(c1cn(CCNC(C2CCO2)=O)nn1)=O c1(C(=O)NCC(CC)NC(C2CSCN2C(C)=O)=O)sc(C)cc1C N1(C(C)=O)CC2CC2C1C(=O)NC1CCOCC1NC(c1cc(F)n[nH]1)=O CCC(C)(CNC(c1ccon1)=O)C(=O)NC1CCCN(CC)C1 c1(CC)cc([N+](=O)[O-])ccc1NC1CCC2CN(C(=O)C3=NOCC3)CC2C1 Cc1cc(C(N2CCN(C(=O)C(C)O)C(CC(F)F)C2)=O)ccc1C1CC1 N1(C(c2ncn(C)n2)=O)CC(CNC(=O)C=Cc2ccncn2)C(C(F)(F)F)C1 CONC(=O)C(=O)N1CC(O)CC1CC(=O)NCC1(C)CC(C)C1 CC(=O)C(C)CC(C)C(=O)NCc1n[nH]cc1C(=O)NCc1snnc1C C1(O)(C(C)CNC(=O)Cn2nccn2)CCN(C(=O)CCC2NC(=O)NC2=O)C1 c1(CCC)ccc(C(=O)NC2C=CCN(C(c3cn(CCC)nc3C)=O)C2)cc1 C1(NC(c2c(CCC)nns2)=O)CN(C(c2ccccc2Cl)=O)CCC1C C(CC(O)CCO)NC(C(C1CC1)NC(C1CCC(CO)CC1)=O)=O C1(S(C)=O)(CNC(C(=O)N(C(C(C)C)CN(C)C)C)=O)CCC1 c1(C(=O)Oc2c(OC)cc(F)cc2)c[nH]c2c(Cl)cccc12 C1(C(N2C3(CNC(CCC(=O)NC)=O)CCC2CC3)=O)CCC2CC1C2(C)C C1(C(=O)NC(C)CC2CCC2)CC2C=CC1N(C(=O)Cn1cnnc1)C2 c1(C(=O)N)ccc(SC)cc1Cl.n1(COC(C)C)cc(C(N2CCOCC2)(C)C)nn1 CC1CCC(CNC(C2CCC(C)(F)CC2)=O)CN1C(=O)C(=Cc1c[nH]cn1)F c1(C(=O)NC(CCNC(C(C)OCCC=C)=O)C)conc1-c1ccccc1 c1(CC2(C(N3CC(CNC(C45CCC4CC5)=O)C3)=O)CC2)cccc(Br)c1 C1(C)(C(=O)NC(CC)CNC(c2coc(COC)n2)=O)C=CCCC1 c1(C(=O)NC2(CC=C)CN(C(=O)CCc3cc(OC)no3)C2)ccc(F)nc1 CC1OC(=O)NC1C(=O)NCC1CCCC1NC(=O)CCC1CC1(C)C C1(NC(C(c2ccccc2F)C)=O)CN(C(=O)CCP(C)(C)=O)CCC1C N1(C(c2c(C)con2)=O)CCN(CC(C)NC(=O)CCC2CCC(=O)N2)CC1 CC1(CNC(C2(c3ccccc3)CCCCO2)=O)CCCN1C(C1COCO1)=O CC1CCc2onc(CNC(c3c(F)ccc(OC(F)F)c3F)=O)c2C1 C1(NC(CCc2onc(C)n2)=O)CN(C(=O)Cn2cc(Cl)cn2)CCC1C c1(OC(CCC(C)C2CC2)=O)ccnc(OCC(F)F)c1 C1(C)(C(=O)NCC(CC(=O)NCCCC2CC(C)C2)OC)CCC(O)CC1 C#CC1(CNC(=O)C=CC2CCCN2C(c2ccc(C)cc2)=O)CCOCC1 c1(OCC)ccc(N)c(C(=O)NCCC2CN(C(=O)CC(C)CF)C2)c1 C#Cc1ccc(Cl)c(C(N2CC(NC(C3CCn4cncc4C3)=O)C(O)C2)=O)c1 c1(OC)cc(F)c(F)c(-c2cn3cnc(C(=O)NCc4ccncc4)c3s2)c1F c1(C(C)N(C(c2sccc2I)C(=O)NCC2CC2)C)cccc2ccccc12 c1(C2C(C(=O)OCC(=O)NC3CC(CC)C3)C2)ccn(C)c1 N1(C(CCCC(C)C)=O)CCC2CN(C(=O)CC3=NNC(=O)C3)CC12 Cc1ccc(F)cc1-c1nc(-c2cccc(Cl)c2)nn1C1CCCOC1 Cn1cc(C(=O)NCC2CCN2C(c2ocnc2-c2ccccc2)=O)nc1O C(C1c2ccccc2CCN1c1ccncc1[N+](=O)[O-])NC(=O)C1=CCSC1 Cc1cc(N(C2CNCCOC2)C(c2ccoc2)=O)n2nc(C)cc2n1 CCC(CC(C)C)C(=O)NCC(CCOC)NC(C1CC(SC)C1)=O c1(N(CCCC)C(=O)NCC23COCC2C3)ccc(C)cc1 CCCC(C)(O)C(=O)NCCN(C)C(c1ccc(-c2ccc(C(F)F)o2)cc1)=O CN1CCC(C(=O)N(C2CCCCC2)CCNC(c2cnc(S)nc2)=O)C1=O C1(NC(=O)C(=O)N=c2[nH]ncs2)CCC2CN(Cc3ccccc3)CC2C1 n1(CC)cc(Br)c(CC(=O)NCCCCC(C)NC(C23CC(O)C2C3)=O)n1 C1(CN(C(=O)Cc2cc[nH]n2)C)CN(C(c2cc[n+]([O-])cc2)=O)CC12CC2 Cc1nnc2n1CCC2(C)C(=O)NC1CN(C(c2csc(C#N)c2)=O)CC1C N1(C(CC2(SC)CC2)=O)CC(CNC(c2cccnc2N(C)C)=O)C2(CCC2)C1 N1(C(=O)CCCOc2ccc(F)cc2)CC2CCN(C(=O)Cc3ccns3)C2C1 C(=O)(C(O)C(C)(C)C)NC(C1(O)CN(C(=O)CCCc2c(F)cccc2F)C1)C C1(OCC(=O)NCCCN(C)C(c2occc2Cl)=O)CCC(N=[N+]=[N-])CC1 CC1OC2(CO)CC1(C(=O)NCC(F)CNC(=O)COC1CCCC1)C2 Cc1nc(C(=O)NC(Cc2ccco2)C(=O)NC(C)C(C)(C)O)sc1C C#CCCN=C(NCC1CCC(=O)NC1)NC1CCN(CC)C1 CCCC(CC)N=c1[nH]c(=NC(C)c2nc(CN(C)C)cs2)c2cc(Cl)ccc2[nH]1 c1(C(=O)NC(C(C)C)CNC(=O)C2=CCCC2)ncn2c1CCCC2 C(=O)(CCCC(=O)C1CC1)NCC(CNC(=O)Cc1cccnc1)CO n1(C(=O)NC2CC(OC(F)(F)F)C2)cc(C2(O)CC2)nn1 c1(OCC#C)cc(CN2CC(OC)CC2CO)c(OC)c(Br)c1 c1(C(N2C(CCCNC(COC(CC)C)=O)CCC2)=O)cccc([N+](=O)[O-])c1Cl c1(OC)cc(C(=O)N(C(C)C)Cc2cc(Br)ccc2F)c(NC(=O)C(F)Br)cn1 CN1CCN(C(=O)CSCCC#N)CC1CNC(=O)C(O)CC1CCCC1 c1(C(N2CC(OC)C(NC(=O)C(C)C3CC3)C2)=O)cnn2c1CC(F)(F)C2 c1(C(=O)NC(C2(O)CCN(C(=O)CCC3(C)CC3)C2)C)cc(C(F)F)ccn1 CP(C)(=O)C(CC(=O)NCC(CO)NC(c1c[nH]ccc1=O)=O)P(C)(C)=O CC1CCC2(CCO2)N(CC2NC(=O)CC2(C)C)C1 CC(C)(C)C(=O)CCC(=O)NC1CC(OCC(N2CC3CCC2C3)=O)C1 c1(CNC(C2CC(F)C2)=O)ccccc1CNc1ncccn1 Cc1ccc(CNC(C2(CC(N3C(C)C(C)CCC3)=O)CCC2)=O)c(O)c1.N(C)C C1(CNC(CC2(OC)CC2)=O)CN(C)CCN1C(c1cnc(C)nc1C)=O c1(C(N(CC(C)(C)NC(c2cc(C)sc2N)=O)C)=O)cncc2n[nH]cc12 N1(C(CC23CC(C)(OC2)C3)=O)CC2CCC1C1CN(C(c3ccc(Cl)o3)=O)CC21 N1(C(C(CCSC)O)=O)CC2CCC1C1CN(C(=O)Cc3ccc(Cl)c(F)c3)CC21 C1(NC(C(C)CN2CCCCC2)=O)CN(C(=O)C=CC(=O)N(C)C)CC1F C1(NC(C2(COC)C=CCN2C(=O)C=CC2CCCN2C)=O)CCC(=O)N(C)C1 N1(C(C(CSC)OC)=O)CCC2(CC1)CC2(CO)CNC(=O)COc1ccon1 c1(C(N2CCN(C(c3cscc3C(F)F)=O)C(CCO)C2)=O)cc(O)cc(=O)o1 N1(C(C2CCN(C(C3CC(SC)C3)=O)C2)=O)CCOC(C)C1CO C(C(C)C(C)CC)NC(CC1(C=C)CN(C(=O)CCCC(=C)C)C1)=O C1(NC(c2cc(C)n(C)n2)=O)CC2CCC(C1)N2Cc1cc(C(F)(F)F)on1 CC1(C)CN(C(C23CCCCC2C3)=O)CCC1NC(C1C2C3CCC(C3)C12)=O N1(C(CC(C)SC)=O)CCSCC1CCNC(=O)Cn1nccn1 Cc1ccn(C)c1C(=O)NC1CCN(C(c2ccon2)=O)C1Cc1ccccc1 Cc1cc(C(N2CC(C)CCC2CNC(=O)CCc2csc(C)n2)=O)nc(C)c1 c1(C(N(CC(C)NC(=O)C(=Cc2cnc[nH]2)C)C)=O)cc(C(C)C)[nH]c1C(C)C C12(CNC(CCCN(C)C)=O)CCC1CCN2C(=O)Cc1cccnc1Cl C=C1CCN(C(=O)C(CC)CC=CC)C(C(=O)NC(C(O)CO)C2CC2)C1 c1(NCCCN(C(=O)C=Cc2cccc(Cl)c2)C)c(C#N)c(=O)n(C)c(=O)n1C N1(C(C(C)SC)=O)CCC(CF)(NC(=O)CCc2cnc(C3CCC3)o2)C1 CC1(C(=O)NC2CC2NC(c2sccc2CC#N)=O)CCCC1(F)F c1(OC)ncnc(C(=O)NC(CNC(c2cn(C)nc2C)=O)C(C)C(C)C)c1F c1(C(N(C)CCNC(C2CCCCC(C)(C)C2)=O)=O)cc(N=S(C)(C)=O)ccn1 C(=O)(C(CNC(=O)C(C)CCOC)C(C)C)N(CCC)CC1CC1 c1(C(=O)NCCC(C)NC(C2CCCC(C)O2)=O)cnn2c1CC(F)(F)C2 S(=O)(=O)(c1cnn2ccc(N3CCCC(C)C3)nc12)N(C)CC1C(OC)COC1 C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)(NC(c2ccc(C)o2)=O)C1 Cc1ncc(C(N2CCC(NC(=O)C(c3ccccc3)F)C2C(C)C)=O)n1C Cc1cccc(CN(CC(C2CCCC2)C)CCc2ccccn2)c1C C12(C(N(C(CNC(C(C)NC(C)(C)C)=O)(C)C)C)=O)CC3CC(C1)CC(C)(C3)C2 CCCCC(C)(c1nnnn1C1CCCC1)NCCC(N)=O C1(NC(C2CCCCC2)=O)CN(C(c2cn3ccsc3n2)=O)CCC12CCC2 N1(C(c2c(CC)nns2)=O)CCC(NC(c2snnc2C)=O)C(O)C1 c1(C(=O)OCC)cccc(C(=O)NC2(C)CC(NC(=O)CC(C)(C)O)C2)n1 C(=O)(C(C)S(C)(=O)=O)N.C(C(C)(C)C(=O)N(CC1=NOC(C)C1)C)OC CN1CCCC1C1CCCN1CC(C1(C(=O)O)CC(C(=O)O)C1)=O C(CCCCCO)NC(C1N(C(CCCOC(C)C)=O)CC=C1)=O C(=O)(CCC(=O)N1CCC(CNC(C23CC(C2)C(C(F)(F)F)O3)=O)C1)NC c1(C(N(C)CC2C3CN(C(C4CCC(CC)O4)=O)CC32)=O)ccn2nnnc2c1 CN1CCCC(F)(C(=O)NCC(C2CCN(C(=O)Cc3cccs3)CC2)(C)O)C1 c1(C(N(C(CN(C(c2ncc(CC)cn2)=O)C)C)C)=O)cc2ccc(C)cc2[nH]1 N1(C(CCC#N)=O)CC2CC2(NC(c2cc(-c3ccccn3)c[nH]2)=O)C1 C1(C(=O)OC)CC2(CC2)CN1C(C1(O)CCN(C(C2CC(C)CO2)=O)C1)=O c1(C(N(C2CN(C(=O)NC3(SC)CC3)C2)C)=O)ccc(C#N)o1 N1(C(c2cnc(CC)s2)=O)CCC(CO)(NC(=O)C(C)n2ccnn2)CC1 c1(C(N2CCC3CN(C(CCC(=C)C)=O)C3C2)=O)ccc2c(c1)OC(C)(C)O2 C1(N(C)C)(C(=O)NCCCC2CCN(C(C3CC3[N+](=O)[O-])=O)CC2)CCCOC1 c1(NC(c2cn(C)c(C(F)F)n2)=O)ccc(C(=O)O)cc1O Cc1nc(NCC2CC(CNC(c3nc(C)sc3C)=O)CO2)c(C)c(O)n1 N1(C(CC(CCCC)CC)=O)CCC2(CCCCC2NC(c2c[nH]c(C)c2)=O)C1 N1(C(C2C=C(C)CS2)=O)CCC(NC(c2cc(C(C)C)no2)=O)C(C)C1 N1(C(CN2CC(C)C2)=O)CC(NC(=O)C(O)c2ccsc2)CC12CCCCCC2 C1(CNC(C(C2N(C(c3cc(OC)n[nH]3)=O)CCC2)(C)C)=O)CC2CCC1O2 C#CCC(C)C(=O)NC(C)Cn1cc(CNC(c2cnc(OC)nc2)=O)nn1 N1(C(CCOCCCOC)=O)CC(CNC(=O)C(C)CO)C(F)(CO)C1 N1(C(=O)NCc2noc3c2COCC3)CCC2(CC1)C(O)CC2O C=CCC(F)(F)C(=O)NCC(C)CC(=O)NCC(=O)NC c1(N2CCn3c(CO)nnc3C2)[nH]c(=NC2CCC3CCC23)nc2sccc12 c1(OC)c(C(=O)NC(CNC(C2(CCCCO)CCCC2)=O)CO)cccc1F CC(C)(CC(F)F)C(=O)NCCCNC(=O)CC1CCCC2(CCC2)O1 N1(C(C2CCC(=C)CC2)=O)CCCCC(NC(C2CCCC(=O)N2C)=O)CC1 C1(O)(COC(C)=O)CCN(C(C2COCCC2NC(C2(OC)CC2)=O)=O)CC1 C(=O)(C1CCCn2nccc21)NCC1N(C(c2c(C)ccnc2)=O)CCN(C)C1 c1(C(=O)NC(C2CCN(Cc3ccc(NC(N)=O)cc3)CC2)C)cccc(F)c1 C(N=c1[nH]c2c(c(=NC(C)C3(CO)CC3)[nH]1)CCCC2)c1c(C)occ1 c1(C(N2CCCC(F)(CNC(c3ccnc(Br)c3)=O)C2)=O)ccc2ncnn2c1 N1(C(C2(C)CC3CC3C2)=O)CC2CCN(C(c3ccc(S(N)(=O)=O)o3)=O)CC2C1 Cc1cc(CCC(=O)NC(C)CC(C)NC(c2cnc(O)o2)=O)cc(C)c1 N1(C(C(C)=CC2CC2)=O)CC2(CC(NC(c3c(C(F)(F)F)cccc3F)=O)C2)C1 c1(OCC)c(C(=O)NCC(CSC)OC)cc(C(=O)NCC)cc1OC c1(C(N)=O)ccc(Cl)c(NC(=O)NC2CCCC2n2cccc2)c1 C1(OC)CC2CCC1(C(N1CCCC(C(N3CCN(CCO)C(C)C3)=O)CC1)=O)C2 N1(C(c2c(CC)ocn2)=O)CC(NC(c2c[nH]cc2Br)=O)CCC1C CC1(C#CC(=O)N2Cc3ccccc3CC2C(N2CC(O)C(O)C2)=O)CCCO1 Cc1c(-c2nc(-c3ccc4c(c3)NCCC4)no2)cccc1[N+](=O)[O-] N1(C(C(CC=C)OC)=O)CCC(C(=O)N(C2CCO2)CC=C)C(O)C1 CCCCC(CNC(=O)C(C1CC1)C1CC1)NC(=O)Cn1cnc(C(N)=O)n1 N1(CC)CC(C(N2CCC(C)(NC(c3ncccc3Cl)=O)C2)=O)NC1=O C1(NC(C2CC2(Cl)Cl)=O)C2CC3C(C2)C13C(=O)NCC1(F)CCOC1 C(CCC(=O)NCCCNC(c1cc(-c2ccc(Cl)s2)[nH]n1)=O)=CCC=C Cc1nc2ccccc2c(C)c1CC(N1CCC1c1cccc(Br)c1)=O N1(C(=O)OC)CCN(C(=O)C(Cc2cc[nH]n2)NC(C2C(C)C2C)=O)CC1 C(C1CCCCCC1)=CC(N1CCCC(CN(C(c2ccc(CC)o2)=O)C)C1)=O N1(c2nnc(C(C)C)o2)CCC2(CCC2)C(NC(=O)CCc2ncc[nH]2)C1 N1(C(=O)NCC(c2cccc(F)c2)C)CC2(C1)OCC1CC21 c1(OC)ccc(O)cc1C(N1CCC(C)(C(=O)Nc2cnc(F)cc2C)C1)=O CC1OC2(C)CC1(C(=O)NCC1CCC(NC(c3ccnnc3O)=O)CC1)C2 CCCC(C(=O)NCC1(NC(c2cncn2CC)=O)CCC1)c1cccc(Cl)c1 C1(CC(=O)NCC(C)CN(C)C(c2ccccc2Br)=O)CCC(=O)NC1 C12(CC(=O)NCCCCCC)CCC1CN(C(=O)C(n1nccc1C)C)C2 N1(C(COc2cc(C)on2)=O)CCC(C)C(CC(N2Cc3c[nH]nc3C2)=O)C1 c1(NC(CC(=O)N(C2CN(C(=O)C=CC(C)C)CC2F)C)=O)cc(Cl)cc(Cl)c1 CC(C(=O)NCC1(O)CCCN(C(=O)CCSc2ccc(F)cc2)C1)C(C)(F)F C1(C)(CNC(Cc2c(C)cncc2)=O)CCCN(C(C2OCCCC2(C)C)=O)C1 C(=O)(CS(=O)CC)NCC1(CCNC(c2nc(CCCCC)sc2)=O)CC1 c1(C(=O)NC2CC(NC(CSCC(=O)Nc3ccccn3)=O)C2)cnncc1O Cn1c(NC(N2CCC3(CCC(=O)NC3)C2)=O)nc2cccc(Br)c12 C1(CNC(C2C(CCOC)C2)=O)C(C2CC2)CCN1C(C1CN2CCN1CC2)=O Cc1ccc(-c2nc(CO)nn2-c2ccnc(O)c2)cc1[N+](=O)[O-] Cc1cnc(NC2CCC3CC3CC2)c(S(=O)(=O)NC2CCC(C)CC2)c1 N1(C(Cc2ccc(C(=O)OC)nc2)=O)CC2(C1)CN(C(=O)C=Cc1cnn(C)c1)C2 Cn1ccc(=NC(=O)N=c2nc(Cl)[nH]cc2-c2ccc(N3CCCC3)cc2Cl)[nH]1 c1(C(=O)NC2CC(F)(CNC(c3c(OC)n[nH]c3)=O)C2)c(C)cccc1C C1(NC(=O)CC2CCCCN(CC=CC3CCOCC3)C2)CCOCC12CCC2 Cc1ccc(C(N)=O)cc1C(=O)NC1(CN(C(=O)C(CC(C)C)N(C)C)C)CC1 C1(C(=O)NC2C(SC)CCC2)CC2CC1CN(C(=O)C=Cc1cocn1)C2 c1(NC(C(C(C)NC(C2(CC=C)CC2)=O)C)=O)ccn2nccc2c1 C1(N(C(CC(c2cccc(OC)c2)C)=O)C)CCCCN(C(=O)CCC(C)C)C1 c1(NC(C2C=CC(NC(=O)C(F)F)C2)=O)cc2nccn2cn1 C12(CN(C3(C(C)(F)F)CC3)CC)CCCN(C(=O)COc3ccccc3)C1C2 c1(OC)cnc(C(=O)NC2CC(CO)N(C(=O)CCC(N)=O)C2)c(F)c1 c1(SC)ccc(OC(C)C(=O)NC(C2C=CC(CNC(=O)CC(C)F)C2)=O)cc1 C#CC1(N)CCCOC1.C(=O)(CCCN(C(=O)COc1cccnc1)C)OC O=C(N=c1ccn(Cc2ccc(F)cc2F)[nH]1)NC1CCN(CCO)C(=O)C1 c1(CC(=O)NCC2(F)CC(NC(c3csc(Cl)c3)=O)C2)ccc([N+](=O)[O-])cc1F CON(Cc1ccccc1)C(=O)C(Cc1ccco1)NC(=O)C(=O)NOC c1(C(=O)NC2CCC(NC(C(c3ccc(Cl)cc3)CC)=O)C2)nn(C)c(C)c1Cl CSC1=C(C(=O)NCC(C)CNC(c2ccc(C)c(C#N)c2)=O)CCCC1 C1(CSCC(=O)OCCOCCc2ccco2)CCC(=O)N1 C1(CCC)CCCN(C(=O)C(O)CCCNC(C2(CO)CCC2)=O)CC1 Cc1cc(C(=O)NCC2CC(C)N(C(=O)C(C)NC=O)C2)c(N)c(Cl)c1 N1(CC2C(C(N(CCNC(=O)CC3(O)CCC3)CC)=O)C2)CCNC(=O)C1 N1(C(C2C(C=C)OCC2)=O)CC2CCCC(CNC(c3nc(O)sc3C)=O)C2C1 C1(NC(C)CCC#N)CCCC(N)C1.C=C(C)C=O C1(C(=O)NCc2ccc(Br)c(F)c2)CC2CCC1N(C(C1CCCS1)=O)C2 N1(C(=O)OCC)CC2(CCN(CCCC34CCC(CC3)OC4)CC2)CC1C CN1CC(NC(=O)CC2(C)CCN2C(=O)C(F)CC2CCOC2)CC1CO C1(CCC)CCC(C(=O)NCCNC(=O)C(CC)N2CCCC2=O)CC1 c1(C(N(CCCNC(=O)CCN2CCCC2=O)C)=O)ncsc1S(N)(=O)=O Cc1nc(Cl)ccc1CC(N1CCC(NC(=O)Cc2nncn2C)C12CC2)=O c1(CNC(C(=O)N(C(COC)(C)C)C)=O)nc(C(C)(C)C)ns1 c1(CC(=O)NCC(CNC(c2ccc(CCC)[nH]2)=O)CO)ccc(S(C)=O)cc1 N1(C(c2cc(C)n(C(C)(C)C)n2)=O)CC2C(NC(=O)C(O)CF)CS(=O)(=O)C2C1 c1(C(N2C(CNC(C(COC)(C)OC)=O)COCC2)=O)ccc(Cl)c(F)c1 c1(SCC(CC)(c2ccccn2)NCC2CC2)ccccc1-c1ccccn1.SCC C(CC(O)C(C)C)NC(C1CC(CNC(C2(CC#C)CCOC2)=O)C1)=O C1(CNC(c2n(CC)c(O)nc2)=O)(NC(=O)CN2CCOC2=O)CCCCC1C CCC(C)(C(=O)N1CCCOC(CCNC(c2cnn(CCF)c2)=O)C1)C(N)=O c1(N(CCCC=C)C)ncc(C)cc1S(=O)(=O)NCc1scnc1C C1(C(=O)NC2CN(C(c3cnn(CCOC)c3C)=O)CC2C)CCC2CC1CO2 N1(C(CCC2CCCN(C(c3cc(C)c(O)cc3)=O)C2)=O)CCC(F)(F)C(O)C1 N1(C(CC2(OC)CCCC2)=O)CCCN(C(=O)CC(O)CN(C)C)CC1C N1(C(=O)OC(C)(C)C)CC2C=CC1C(Nc1c(F)cccc1F)C2 C(=O)(C1=C(Cl)CCC(C)C1)NC1C(CNC(Cc2c(OC)cccc2)=O)CCC1 C(C(C)NC(=O)C(C)(C)C1CCOCC1)(C(C)C)NC(CSCCC)=O C(=O)(N=c1cc(CC)n(C)[nH]1)C1CN(C(CCCC#C)=O)CC12CNC2 CC1CCCC1(C(=O)NCC1CC(O)C(O)C1)NC(c1ccccc1O)=O N1(C(CC(c2ccc(-c3ccn(C)n3)s2)C2CC2)=O)CCC(O)CC12CC2 C1(CNC(C2C(=C)C2)=O)CN(C(c2cnn(C3CC3(F)F)c2)=O)CCO1 C(=O)(C1CCCn2cncc21)N(CCNC(CC(C)CCc1ccccc1)=O)C N1(C(N(C)C)=O)CCCc2cc(NS(=O)(=O)c3cc(F)ccc3Br)ccc21 N1(CCNC(C2CC(O)C2)=O)CCCC(CC2CC2)CC1.C1(C2(N)CC2)CCCO1 c1(OC)ccc(Br)c(CCNc2cc(Br)c[nH]2)c1F.c12ncc(s1)CC(=O)N2 c1(OCC)ncncc1NC(C1(C)CCN(C(=O)C=C=C(C)C)C1)=O CC(C)C(O)C(C)C(=O)N1CCCC(CN(C)C(c2cc(C(C)C)cnc2O)=O)C1 c1(CNC(=O)NCCCCS(C)=O)ccc(Br)cc1F C#CC1CCN(C(C2CCN(C(=O)C(=O)C(C)C)C2CC)=O)CC1 C1(CC=CC)CCCN(C(CC2(C#N)CC2)C(=O)NC)C1 C(C(C)(C)C1=CCOCC1)C(c1cccc(-n2cc(CC(CC)(C)O)nn2)c1)=O C12(C(=O)NCCCOC(C)C)COC(C1)C(NC(C1CCC1C)=O)C2 N1(C(c2cccc(OCC)c2)=O)CC(NC(=O)CN2CCCC2)CC1(C)CC C#Cc1ccc(CC(=O)NC2CCN(C(C3CC(CF)C3)=O)CC2C)cc1 c1(N(C)C)cccnc1C(=O)NCC1CC(NC(C2CCC(F)(F)C2)=O)C1 N1(C(c2cnc(CC)nc2O)=O)CCCCCC(NC(C2(CO)CCCO2)=O)C1 N1(C(CCC=C(C)C)=O)CC2CS(=O)(=O)CC2(NC(=O)CCc2cc(C)no2)C1 N1(C(CC(C=C)C)=O)CCC(NC(C23CC(C(F)(F)F)(CO2)C3)=O)C(F)C1 C(=O)(CC(C)P(C)(C)=O)NCCCN(C(CCN(C(CCC)C)C)=O)C Cc1ccc(-n2nc(C3CC3C)nc2C(C)CCN(C)C)cc1C S(=O)(=O)(c1cc(-c2ccc(C=CC)cc2)c(C)cc1C)N(CCOCC)CCO c1(C(=O)NC(CNC(C2(COC)CC2)=O)C2CCC2)ccc(O)cc1 C1(NC(C2N(C(C(C)CC3CC3)=O)CC(F)C2)=O)CC2C=CCC(C1)C2 N1(C(CCC2N(C(c3c(C)oc(CO)c3)=O)CCC2)=O)CC2CC3CC2C1C3 C(=O)(CC(C)(C)C(C)=O)NC(CC)CCC(=O)NC1CC(C)(OC)C1(C)C C1(NC(CS(CC)(=O)=O)=O)CC2CCCC(C1)N2Cc1cccc(CC(=O)O)c1 C(=O)(C1CCCc2c[nH]nc21)NCCCCN(C(C=CSC)=O)C c1(CNC2CCN(CC(C3CC3)NC(C(=O)OC)=O)C2)cccc2nonc12 Cc1c(C(=O)NCC2CC2NC(=O)C(CC#N)C2CC2)oc2c(C)cccc12 C(=O)(C1=CCCCO1)NC(CC(C)C)CNC(c1cncc(C(C)C)c1)=O C12CCCN(C1)C(=O)C(F)C1CC(C1)O2.C1(C(CCC)=O)CC(C)(O)C1 N1(C(c2cn(CC)nn2)=O)CC2(CC2)CC1CNC(c1nccc(Cl)c1Cl)=O C(=O)(C(C)(C)CNC(=O)CC1CC2(CC2)CO1)NCC=C c1(C(=O)NC2CN(C(CCNC(=O)NC)=O)C3C2C3)cc(N)cc(F)c1 Cc1cnsc1C(=O)N(CCC(C)NC(c1[nH]ccc1-c1cccs1)=O)C C1(CNC(C(C2CC=CCC2)NC(c2nocc2Cl)=O)=O)CC2(CC2)C(=O)O1 C1(C(=O)NC(C#C)(C)C)CCN(C(c2cc3ccncc3[nH]2)=O)C12CCC2 C1(NC(=O)CNC(c2cccnc2)=O)CCN(C(c2cnc(O)o2)=O)CC1CO C1(CC(N2C(CNC(c3cc(O)no3)=O)CC2)=O)COC(=O)C1 C1(N(C)C(c2cnn(C(F)F)c2)=O)CCCCC1N(C(=O)CSCC(F)(F)F)C C1(CC(N2CC(OCCOC)C2)=O)CC(C2CC2)C1.c12cc(on1)NC2=O N1(CCC(=O)N(C2CCN(C(c3ccc(NC)cc3)=O)C2)CC)CCCCC1=O Cn1ccc(C(N2CCN(C(C3CC(F)C3)=O)CC2)=O)cc1=O C1(O)(CN(C)C(C2CC2Cl)=O)CCN(C(c2cc(N)ccn2)=O)CC1 c1(COC)cccc(C(N2CCOCC2C)C(=O)NC2CCOCC2)c1.C1(C)CC1 CCCC(F)C(=O)N(C)CCOCCC(=O)NCC(CSC)OC C1(NC(c2c(C)nc(C)s2)=O)CCCC12CN(C(c1nocc1C)=O)C2 Cn1cc(C(=O)NCCN(C(=O)CC2CCCC2(F)F)C2CC2)c(C(F)F)n1 C(CC(C)(C)C(=O)NCC(O)(CO)CO)NC(C(C=C)C)=O C1(CC(=O)NC(C#C)CC2CCCC2)(NC(c2cc[nH]c(=N)n2)=O)CCCCC1 CCCC(CCCNC(c1cc(F)n[nH]1)=O)NC(=O)Cn1nccn1 N1(C(C(CC=CC)CC)=O)C2CCC1CN(C(=O)CCC(F)F)C2 C(=O)(C(F)(F)C1CC1=O)N(CCNC(C1C(OC)C1)=O)C c1(OC)cccc2cc(C(=O)NC(C)CN(C)C(c3ccc(C)cc3Cl)=O)oc12 C(C)(C(=O)NNC(=O)CNC1CCCCC1)SC N1(C(c2c(C)oc(Cl)n2)=O)CCC2(CC1)CN(C(C1CC(F)C(=O)N1)=O)CCO2 C(=O)(C(C)CCCC(C)C)NC1(C(=O)NCC2(CO)CC2)C(C)CCC1 Cc1cc(C(N2CCN(C(=O)C(C)CN(C)C)C(C(F)F)C2)=O)cnc1C C1(NC(CCC(C)C)=O)CN(C(C2COCCN2C)=O)CCC1O c1(NC(=O)NCC2OCCN(C(CC(C=C)(C)O)=O)C2)cccc2cnn(C)c12 C1(C(=O)NCC(CC(=O)NC(C)C(C)(C)CO)C2CCC2)Cc2nccn2C1 c1cnc(S)n1C.Cc1ccsc1-c1cccs1.C12CC(C1)NC(=O)N2 Cc1cn(C(C)C(=O)Nc2ccc(F)cc2F)[nH]c1=NC(=O)C1CCS(=O)(=O)C1 Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCCCC1NC(c1cn[nH]c1)=O Cc1cnc(C(N2CCC2CNC(=O)C(C2CCOCC2)O)=O)cn1 N1(c2ccc(C(C)=O)cn2)CCC2CC(NC(C3CCOC3)=O)CCC2C1 c1(C(=O)NCCCOCCCNC(CSCCC=C)=O)ccn(C(C)CC)n1 N1(C(CC(C)N(C)C)=O)CCOC2CN(C(c3coc(C(N)=O)c3)=O)CC12 C(=O)(C(CCC1CCCOC1)N1CCSCC1c1nc(C)cs1)NC(CC)(C)C C1(CNC(C(c2cccc(C)c2)O)=O)Cc2ccccc2CN1C(=O)CC(F)F N1(C(C)C(=O)NC2CCCC2NC(=O)CCCN2CCOCC2)CCCCCC1 N1(C(c2cc(COC)no2)=O)CCCCC1CC(N1CC(C(C)C)C1)=O C1(C(=O)NCC(C)NC(c2ccn3nccc3n2)=O)CN=C2N=CNN2C1 C1(CN(C)C(c2ccns2)=O)CCN(C(c2ccn(C(C)(C)C)c2)=O)C1 C(CCCC(CO)NC(C1CCCS1(=O)=O)=O)NC(CC(CC)OC)=O c1(C(=O)NCCC2CCCN(C(=O)CSC3CC3)C2)nccn2ccnc12 CC1(C)CC(C)(CNC(C2Cc3nccnc3C2)=O)CN1C(=O)CC(=O)N(C)C Cc1c(Br)ccc(C(N2CCN(C(c3cc(Cl)cc(Br)c3F)=O)C3CC23)=O)c1F c1(C(N(C)CC2CN(C(=O)CSC3CC3)C2)=O)ccc(S(C)(=O)=O)cc1 C1(C(=O)NC2(C(COC)C)COC2)CN(C(=O)OC(C)(C)C)CC(C)(C)C1 N1(C(CSC(C)(C)C)=O)CCC2CN(C(c3sc(N(C)C)nc3Cl)=O)CCC2C1 C=C1COc2c(C(=O)NCC3CCN(C(=O)CCF)CC3(F)F)cnn2C1 Cc1cc(Br)cc2cc(CNCCOCc3ccccc3)[nH]c12 C1(C(N(C)CC2CCN(C(C3CC4C=CC3C4)=O)C2)=O)CCc2nnc(O)n2C1 n1(CC)cc(C(=O)C(=O)NCC2(O)CN(C(c3ccn(C4CC4)n3)=O)C2)cn1 Cc1cc(C(C)C)ccc1NC(C12CC(C1)N(C(=O)Cc1cn(C)nc1C)C2)=O c1(C(=O)Nc2cc[nH]n2)cc2ccc(-c3cccc(F)c3C(F)(F)F)cc2[nH]1 C1(NC(C(CC)C)=O)CC12CCC(NC(c1c[nH]cc(Cl)c1=O)=O)CC2 c1(C(=O)NCC2CCC(NC(C3(C)ON=C(C)C3)=O)C2)cnc2c(c1)CCOC2 CCC(C)C(=O)C(=O)N1CC(O)C(O)C1CNC(=O)CC12CCC(CC1)C2 C(=O)(CCC(N)CCC(=O)OC(C)(C)C)OC.C12CC3CCC(C1)N3C2=O c1(C(=O)NCCN(C(=O)C(C)(C)C2CC2)CCC)cc(C)cc2c[nH]nc12 CC1(C)CC(C(=O)NC2CC3CCC2O3)CCN1C(C1C2(CC2)C12CC2)=O N1(C(CCNC(COCCC#C)=O)=O)CC(C)(CNC(=O)CCC2CC2OCC)C1 Cc1nc2cc(C(=O)NC3CC4CCC3(NC(=O)CNC(N)=O)C4)ccc2s1 c1(NC(C2C(C(=O)NCc3ccc(OCC#C)cc3)C2)=O)cc(Br)cc(C#N)c1 C1(CCC)COCCN1C(c1cnc(C)cn1)C(=O)NC1CC1 C1(C(=O)NC(c2nc[nH]n2)C)(NC(C2(c3cc[nH]n3)CC2)=O)CC(O)C1 C1(C(C)(C)CNC(=O)CC23CCCC2C3)CCCN1C(=O)Cc1csc(NC)n1 c1(NC(=O)CN2CCNC2=O)nc(C(c2ccncc2)=O)n[nH]1 C1(NC(=O)NCCc2cc(-c3noc(C4CC4)n3)on2)CCC(O)CC1 c1(CC(=O)OC)ccnc(N(C2CCCN(C(c3ccc(Cl)nc3)=O)C2)C)n1 O=[N+]([O-])c1cc(F)ccc1CNCC1(Nc2ccc(N3CCCC3)cc2)CCC1 c1(NC(CC#N)=O)cccc(NC(c2ccc(-c3cccs3)[nH]2)=O)c1 c1(C(=O)NCC(CC)NC(=O)CSc2cccc(OC)c2)ccc(N)c(N)n1 c1(C(=O)NCc2c(C)noc2)cc2c(o1)CN(C(=O)OC(C)(C)C)CC2 c1(C(N(CC(C)(C)NC(C2C(CC)CCC2)=O)C)=O)ccc(OC)nn1 c1(C(N2CCC(CC=C)C2)C(=O)NC(C)(C)C)cc2cccnc2s1 C1(C(N2C(C)CC2)=O)CC12CC(NC(=O)CC1(C)CCCCC1)C2 c1(-c2cc(CNC(=O)NC3CCC(C(=O)OC)O3)no2)ccc(F)c(F)c1F N1(C(c2ccc(C#N)cn2)=O)CCCC2(CCCN2C(=O)CCc2cnco2)C1 N1(C(CC2CC(SC)C2)=O)CC(O)(CNC(=O)C2=CCC2)C1 C1(CNC(=O)CC2CCNC2=O)CN(C(C2(c3cccs3)CC2)=O)CC12CCC2 C1(C(=O)NCC(C)C2CCC2)CN(C(C2(CO)CCCCC2)=O)CCC1(C)C C12(CNC(c3cnc(OCC)s3)=O)CC(NC(=O)C(C(C)C)SC)(C1)C(C)O2 N=c1ccc(C(N2CCC(CCNC(=O)CCn3cnnn3)CC2)=O)n[nH]1 C1(NC(c2c(C)noc2C)=O)CCC2CN(C(=O)CC3=NN(C)C(=O)C3)CC2C1 c1(C(=O)NCC2N(C(C(C=C)O)=O)CC=C2)nn(C)c(C(F)(F)F)c1Cl N1(C(CCCC#C)=O)CC(C(C)(C)C)CC(CNC(c2[nH]c(O)nc2C)=O)C1 CCCC(C(=O)NCCN(C(c1csc(C(F)F)c1)=O)CC)N(C)C N1(C(C2C(CNC(C3N(C)CCOC3)=O)CC2)=O)CCC12CCCC2 Cc1nn(-c2ccc(F)cc2)c2sc(C(=O)NCCNC(=O)C(N)=O)cc12 Cc1ccc(F)c(C(C)NC(=O)CC(N)CC2CCCC2)c1 CC1C(NC(=O)C(CC2CCCC2)NC(=O)C(F)C2CCOC2)C1(C)C C#CC1(NC(=O)CSCCNC(=O)CCC(C)CN(C)C)CC(F)(F)C1 C(=O)CCCN(C)N=O.N1(C(c2cccc(CC=C)c2)=O)CCCN(C(N)=O)CC1 N1(C(C2CCN(C(C)=O)C2)=O)CCC2CN(C(c3cccc(=O)o3)=O)C2C1 N1(S(C)(=O)=O)CCC(C#N)(NC(=O)CNC=O)C1.c12cccc(c1)NC(=O)CC2 c1(CC(N2C(CN(C(c3ccccn3)=O)CC)CC2)=O)cnccc1C CC1(C)C(=O)NCC1NC(c1cc(C(F)F)[nH]n1)=O c1(C(C(F)(F)F)(OCC)OC)cn(C2CC=C(C)CC2(S(C)(=O)=O)O)nn1 N1(C(Cn2nc(C)oc2=O)=O)CCCC(NC(C2C=CCCC2)=O)CC1 Cc1c(C(N2CC(O)(CNC(C3CC4CC4C3)=O)C2)=O)sc(Cl)c1Cl N1(c2n(C)ncc2)CCN(C(=O)Nc2ccnn2C2CCCCO2)CC1 C1(CNC(C(CC)OC)=O)(OC)CCOCC1.C1(O)(C(=O)NC)CCCCC1 C(=O)(C1=CS(=O)CCC1)N(C(C)CCNC(=O)COc1ccc(Cl)c(Cl)c1)C Cc1cc(CNC(C2CCC(CNC(C3(C)CCCOC3)=O)C2)=O)ccc1F C1(CC(=O)NC2(CNC(c3c(C)cc(C)o3)=O)CCCCC2)CCCCC12CC2 CN1CCOC(C(=O)NCCOCCC(=O)NCC(C)(C2CC2)C2CC2)C1 Cc1cnc(N2CCN(C(CO)CCC(C)C)CC2)nc1S(C)(=O)=O S(=O)(=O)(c1ccc(F)c2ccccc12)N(CCCC)CC1CCS(=O)(=O)C1(C)C N1(C(C(=O)NCC)=O)CCC2CC2(C(=O)NCc2c(O)cccc2F)CC1 C1(CNC(Cc2c(C)noc2Cl)=O)CN(C(=O)CCS(C)=O)CC1(C)C C1(CCNC(C2CCS(=O)CC2)=O)CCCN(C(C2CCC(C(F)F)CC2)=O)C1 c1(CCC)ccc(CC(=O)NCCOCCNC(=O)CC2CCCCC2C)cc1 C(C)(C)(CC(F)C(=O)NCC1CCCO1)NC(c1cn(C(C)C)nc1)=O CN1CC2(CCN(c3cc(NC4CCN(C(C)(C)C)C4)ncn3)C2)C1 C1(N(C)C)(C(=O)NC2CC(NC(C34CC(CCO3)C4)=O)C2)CCCSC1 N1(C(CSC)=O)CC(CNC(C2COC(C)(C)CO2)=O)OC2(CCC2)C1 C1(C(=O)NC2CC(C)(N)C2)CCc2nccn2CC1.c1(C(C)C(N)=O)cnn(CO)c1 N1(C(CC=CC)=O)CCCC(NC(c2ccc(CC)c(OC)c2)=O)C1C C(C(C)(C)C)N(C)C(C1CC(NC(=O)COCc2cocn2)C1)=O CCCCC(C)C(=O)NCC(CC(=O)NCCOCCCF)O C(=O)(CC(C)CN(C)C)N1CC(CN=[N+]=[N-])(CNC=O)C1.C=CC1CC1 c1(CC)ccc(C(=O)NC(C)CN(C(=O)CCc2ccncc2)CC)s1 Clc1ccc(-n2nc(-c3cccc(N4CCCC4)c3)nc2COC2CCOC2)cn1 CC(C)(CC#N)C(=O)N1CC(CNC(C2CC3C=CC2O3)=O)C(F)(F)C1 c1(C(=O)Nc2scc(C(N(CCC(N)=O)C3CC3)=O)n2)ccc2nc(Cl)ccc2c1 Cc1cc(NC(=O)CC(CC2CC2)NC(=O)C(O)C2CC2)cc(C)c1 C1(CNC(C(N2C(=O)CCC2=O)C)=O)CN(C(=O)CSc2ccncc2)CC1O N1(C(C(C)CN(C)C)=O)CC2CCCC1C2CNC(c1cc2ccsc2n1C)=O C1(CC(C)NC(c2snc(Cl)c2Cl)=O)CCN(C(C2CC3(C2)CC3F)=O)CC1 Cc1cccn2ncc(C(=O)NCCC(C)NC(c3ccn(C)n3)=O)c12 c1(CC)noc(C)c1C(=O)N(CCNC(=O)CSCc1csc(C)n1)CC.C(COC)N N1(C(=O)COc2cccc(C3CCNCC3)c2)CCC(O)(c2ccccn2)C1 C1(C(N2CCC(C(C(=O)N(CC(F)F)CC)F)C2)=O)CCCC1(C)C C1(CNC(C2CCCN(C(C)C)C2)=O)CCN(C(c2cocn2)=O)CC1(F)F CCN=C(NCCCN1CCC1)NCc1ncnn1-c1ccccc1 Cc1nc(CO)ncc1C(N1CC(O)(C(C)NC(C2CCNC2=O)=O)C1)=O C(C(=O)N=c1cc2n([nH]1)CCN(C)C2)n1cc(C(COCCOC)C)nn1 c1(OCC(N2CCN(C(C(=O)NCC)=O)CC2)=O)ccc(C)cc1C C1(C(N2CC(C)(OCC)C2)=O)CN(C(c2scc(C)c2C)=O)CC1(F)F c1(OCC(=O)NC2CC(NC(c3nc(C4CC4)cs3)=O)C(O)C2)cccc(Cl)c1 c1(C(N(CC(CNC(CS(CC)(=O)=O)=O)C)C)=O)cc(C)ccc1[N+](=O)[O-] C1(C(=O)NCC(CC)(C)OC)CNC2(CC2)CO1 n1(CC(=O)NC2C(NC(C3(C(=O)OCC)CC3)=O)CC2)nnnc1C N1(CC2(C(=O)Nc3ccc(C(C)=O)c(O)c3)CC2)CC2CCN(S(C)(=O)=O)C2C1 Cc1nc(NC2CC(CNC(C34CCOC3CCOC4)=O)C2)ncc1Br C(=O)(C(O)C1=CCCCC1)N1CC2C(C(=O)NCC3(C)N(C)C(=O)CC3)(C2)C1 N1(C(Cn2c(C)cc(C(F)F)n2)=O)CCC2(NC(=O)C#CC3CC3)CCCCC12 c1(C(=O)NCC(CC=C)NC(c2ccccc2Cl)=O)ncccc1N=[N+]=[N-] C(C)(C)(CC(F)C(=O)N(C)CC1CCCO1)NC(C(C)C(F)F)=O Cc1cc(=NC2CS(=O)(=O)C23CCOCC3)[nH]c(NC2CCc3c[nH]nc3C2)n1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(C)N(C(=O)Cc1cnn(C(C)C)c1)C C1(N(CCO)CC)CCN(C(=O)CCC(=O)N2CCC(O)CC2)CC1NC(C)=O c1(C(C)C(=O)NCC(=C2CN(c3nccc(C(F)F)n3)C2)F)cccc(F)c1F c1(C(=O)OC)ccc(C(=O)NC2CN(C(c3nocc3Cl)=O)C2)cc1Cl c1(-n2ccc(NC(c3ccc(OC(F)F)cc3)=O)n2)ccc2c(c1)OCO2 c1(OC)cc(Br)cc(C#N)c1.C12CC(=O)CN1C(=O)N2 CC(CC(=O)NCC1(CNC(c2scnc2Cl)=O)CCOCC1)C(C)(C)C N1(C(c2c(C)cc(F)nc2)=O)CC2CC1CCC2NC(C1CN(C)CCO1)=O CC1=C(C(=O)NCC2(NC(c3ccnnc3O)=O)CCOC2)CCCO1 c1(OC)ccc(F)c(C(=O)NC2CCC(C(=O)NCC3CC4C=CC3C4)CC2)c1 c1(OC)cccc(CCC(=O)NCC2(NC(c3cncnc3C)=O)CC2)n1 C(C)(CCCC(=O)N1CC(c2nncs2)C1)NC(C(=CC1CCCC1)C)=O c1(C(=O)NCc2scc(C(=O)NCc3cc(C)ncc3)c2)ccc2c(c1)CC2 Cn1ccc2c(CNc3ccc4c(c3)CNCC4)cccc12 c1(CN2CCCC(NC(c3[nH]cc(C)c3C)=O)C2)nc(O)c2ccccc2n1 CS(=O)(=O)c1ccc(C(=O)NC2CC(O)CN(C(c3ncc(Cl)cc3F)=O)C2)o1 C1(N(C(c2cn(-c3cnn(C)c3)cn2)=O)CC)CCN(C(=O)C(C)(C)SC)CC1 C(C(=O)Nn1nnc(C)c1C)N(C(C)(C)CCCF)CC c1(C(C=CC(=O)NCC(C)NC(c2nnc(S)n2C)=O)=O)cccc(F)c1 CS(=O)(=O)C1CCCC1C(=O)NCC1(F)CC(NC(c2cccc(=S)n2O)=O)C1 c1(C2CCN(C(C(=O)NCC(C3CCCC3)C)=O)C2)ccccc1F C12(NC(=O)CCc3cnc[nH]3)CCCC1N(C(C1CCCCC1)=O)CC2 N1(C(CC(=C)C)=O)CCC2OCCN(C(c3cc(CC)nn3C)=O)C2C1 n1(COC)ccc(C(=O)NC(C)(C)CCNC(=O)C(C)N(C)C(C)=O)n1 N1(CC)CCOC(C(=O)NC(C)CC(C)NC(c2ccc(Cl)s2)=O)C1 C1(C(=O)NCCCNC(=O)OC)CC2CCC(C1)N2C(C1CCC2CC1CO2)=O c1(N(CC(=O)Nc2cccc(C(F)(F)F)c2)C(C)C)sc2c(c1C#N)CCCC2 CCC(C)(CNC(C1COC(CNC(=O)CCC=C(C)C)C1)=O)C(N)=O C1(CC)C(NC(=O)Cc2csc(C)n2)CCCN1C(=O)CC1CC1C(F)(F)F N1(CC)CCN(C(=O)CNC(=O)CNC(C23CCC(C2)OC3C)=O)CC1C N1(C(C2CC=CCC2)=O)CCC2(CC1)CN(S(=O)(=O)C1CC1)C2 C1(CCNC(CCSCC)=O)CN(C(=O)CC2CC(OC(C)(C)C)C2)CC1C N(C1CCc2cccc(NSC(C)(C)C)c21)C(C1=NOC(C)C1)=O c1(NC(C2(O)CCN(C(C(Br)=C(C)C)=O)CC2)C)cc(=O)n(C)c(O)n1 C1(CC)(NC(=O)C=C2CCOCC2)CCN(C(C2CCCC(N(C)C)C2)=O)CC1 C1(NC(CCCOCCOC)=O)CN(C(c2cc(F)cnc2O)=O)CCC1F c1(C(N2CC3(CN(C(c4ccc(Cl)cc4I)=O)C3)C2)=O)cccc([N+](=O)[O-])c1I CCCC(C(O)C(=O)NCCc1nc[nH]n1)NC(=O)C(C)N1CCCC1 C1(N(C(c2c(C)ocn2)=O)C)CCN(C(C2(C(C)(C)O)CC2)=O)CC1 CC1COCC(CNC(=O)C(C)(C)NC(=O)CCOC(C)C)O1 C=CCCCC(=O)NC(C1(O)CCCCC1)C(=O)NCCC1CCOCC1 c1(N(C)CC2CCC(=O)NC2)[nH]c(=NCC2CC(C(F)(F)F)CO2)nc2sccc12 c1(C(=O)NCCNC(C(c2ccc(OC)cc2)CC)=O)ncc2[nH]ncc2n1 C1(CCC(C)(C)NC(=O)COc2ccsn2)CCCCN1C(=O)C1=CCCS1 Cc1ccc(C)c(C(N2CC=CC(NC(=O)Cc3coc(C)n3)C2)=O)n1 O=C(C1=CCCCO1)NCC1C2CC1N(C(=O)CN1CCCCS1(=O)=O)C2 CC(CC(=O)NC1(C)CN(C(C2CCC(C(N)=O)O2)=O)C1)C(F)(F)F CC(C)S(=O)(=O)CC(=O)NCC#CCNC(c1cccc(OCC=C(C)C)c1)=O C1(C(=O)N(C2CN(C(c3coc(-c4cccs4)n3)=O)C2)C)(COC)CCCOC1 CC1CCC(C)(C(=O)NCC(C)(C)NC(c2csc(-c3ccccn3)n2)=O)C1 c1(C(N2C(C)CC(CNC(C3(CCF)CC3)=O)C2)=O)c[nH]c2ccccc12 c1(-c2cn(CC(N3CCC4(CCCO4)CC3)=O)nn2)ccc2nccnc2c1 C1(c2ccccc2)(OC)CC(NC(C2CC2NC(c2c[nH]nc2F)=O)=O)C1 CCC(O)C(F)(F)C(=O)N1CCCC(C)(NC(=O)CCNC(c2ccccn2)=O)C1 N1(C(Cc2n(C)c(S)nn2)=O)CC2CN(C(=O)CC3CCCCC3(F)F)CC2C1 C1(C(N2C3(CNC(CNC(=O)NC)=O)CCC2CC3)=O)CCCCC12CCC2 C(=O)(N=c1[nH]nc(Cl)c2ccccc12)NCC1(OC)CCCSC1 c1(CNC2CC(C)CN(C(C34CC(C3)C4)=O)C2)cc(Cl)c(O)c(Cl)c1 N1(C(c2c(OC)n[nH]c2)=O)CCC(CC(=O)NCC2OCCCC2(C)C)C1(C)C C1(NC(C(C=C)(C)O)=O)CC12CCN(C(=O)CCC(=O)N(C)C)CC2 N#Cc1cc(S(=O)(=O)Nc2cnc(F)cc2C(=O)NC(CO)C2CC2)ccc1Br N1(C(CCNC(=O)NC)=O)CCC(NC(=O)CCc2nc[nH]n2)C(C(C)C)C1 Cn1cc(C#N)cc1C(=O)NCc1cc(C(=O)NCCc2c[nH]nc2O)n[nH]1 N1(Cc2cn(Cc3nc(C(C)(C)C)oc3)nn2)CC(=O)N(CN(C)C)C1=O N1(C(C(c2ccc(Cl)s2)C)=O)CC2(CCC2NC(c2cnc(C(F)F)s2)=O)C1 Cc1nc(Cl)ccc1CC(=O)N(C(CNC(C1(C)CC1(F)Cl)=O)C1CC1)C N1(C(C2C(=C)C2)=O)CCCC(C)(CNC(c2nc(C(F)(F)F)cs2)=O)C1 C(CC(C(C)C)NC(c1ccc(C#N)[nH]1)=O)NC(Cc1nc(C)[nH]n1)=O CCCCC(O)C(=O)N1CC(C(=O)NCCNC(c2cnnn2C)=O)C1 c1(SCC)cncc(C(N2CC(O)CC2CNC(c2sc(C)cc2OC)=O)=O)n1 N1(C(C(C)CC2CCC2)=O)CCOC(C(=O)NC2(C)CCC2)CC1 c1(C(=O)Nc2nccc(CC)c2)ccc(C2=CCCC2)cc1 c1(C(=O)NC(CCc2cccc(OC)c2)C(=O)O)c[nH]c2cncc(Br)c12 Cc1ccc2c(C(=O)N(C)CC3(NC(=O)CC4C=CCCC4)CC3)coc2c1 C1(C)(CN(C)C(C2CCC3(CCC3)O2)=O)CN(c2nnc(C3CC3)s2)CCO1 c1(C(c2nnnn2C2(C)CC2)NC(c2scc(C)n2)C)ccc(N(C)C)nc1 C(CCCC(C)(F)F)(C(=O)OC)N1C(CC)C(CC)CCCC1 c1(C(N2C(C(=O)Nc3cnc(C)nc3C)CCCC2)=O)cnn2ccccc12 N1(C(C2(SC)CCC2)=O)C2CCC1CN(C(c1cnn3ccccc13)=O)C2 C(CN=C(NC(C)C)NCc1ccc(OCC2CC2)cc1)C1(OCC)CCSCC1 CC1N(C(c2ccn(CCNC(c3sccc3C#N)=O)c2)=O)CCCC12CCC2 C12(CNC(CN(CCC)C)=O)CC1CN(C(C1(COC)CC(F)(F)C1)=O)C2 c1(OCC=C)ccc(C(=O)NC(C)(CNC(c2csnn2)=O)CO)cc1OC c1(C(=O)NCC(CNC(CNC(CC)=O)=O)C)cc(Br)cc(F)c1O c1(SC)nc(O)nc(C)c1C(=O)NC(C)CN(C(=O)CC1OCCO1)C N1(C(C2CN(C(c3ccncc3)=O)C2)=O)CCCC(n2nccn2)C1 N1(C(C(C2CCOC2)OC)=O)CC(C)(NC(=O)CCNC(=O)CO)C1 N1(C(c2ccccc2)=O)CC2=C(C1)CN(NC(C13CCC(CC)(CC1)OC3)=O)C2 N1(C(c2sc(Cl)cc2Cl)C(=O)NC(C(=O)OC)C)CCCC2(C1)CC2(F)F N1(C(C(CC)C#N)=O)CCC(CC(N)=O)(N(C(=O)CC2CCCOC2)CC)CC1 CC1NC(=O)CCC1CNC(=O)C(N1CCCC(c2ccc(O)cc2)C1)=O c1(C(=O)NCCCN(C(C2(C#C)CCC2)=O)C2CC2)cc2ccncc2s1 c1(N(CCCC)C2(c3ccccc3F)CC2)nccc(Br)n1 c1(C(=O)NC(C2CCCN(C(c3ccncc3F)=O)C2)C)ccc(F)c(F)c1Cl C(C(C(=O)NC1CC(C(N)=O)C1)NC(=O)CCc1cnn[nH]1)N(C)C C(=O)(C1=CC2CCC(C1)C2)N1CCC(C(C(=O)NC(CCSCC)C)C)CC1 C1(CNC(C(C)NC(=O)C2CC2)=O)CN(C(=O)Cc2ccc(F)cn2)CCC1(C)C c1(C(=O)NCC2(CNC(C3(C)C(C)OCC3)=O)CCC2)ccnc2ccncc12 S(=O)(=O)(c1ccc(NC(C)CN(C)C)cc1Br)NC1(CCOC)CCOCC1 c1(C(n2cc(C3(NC(CC)=O)CCCOC3)nn2)C)ccc2ccccc2c1 c1(C(=O)NCC2(NC(CCN(CCCCC)C)=O)CC2)onc2ccccc12 C1(CNC(=O)CC2C=CCCC2)CCCN(C(=O)CCN2CCCC2)C1 N1(C(c2ccc(C)o2)=O)CCCC(C2CCN(C(C3(F)CCCOC3)=O)CC2)C1 N1(C(CCNC2CN(S(CC)(=O)=O)C2)=O)CC(NC(=O)CC(C)C)CCC1C C12(NC(C3C(C)NCC3)=O)CCC(CC1N)C2 c1(C(=O)NCC2C(NC(CC3(CSC)CC3)=O)C2)ccc([N+](=O)[O-])cc1Cl N1(C(=O)Cc2ccsc2)CC2CC(C1)C2NC(=O)C(F)(F)CN1CCCC1 c1(CC(=O)N(CC(O)CNC(=O)Cc2cc(Cl)cs2)C)cccc(C(F)F)c1 c1(C(=O)N(O)Cc2ccccc2)ccc(-n2c(O)nnc2O)cc1 C1(CN2CC(O)(C(C)(C)CNC(C3CC3c3nc(S)n[nH]3)=O)C2)CC2CC1C1CC21 N1(C(C2N(C(C3(C)CC=CC3)=O)C3C(C2)C3)=O)CCn2cncc2C1 C1(C)(NC(CC=CC=C)=O)CCN(C(=O)COC(C)=O)C1 N1(C(c2c(CC)cc(N)cc2)=O)CCCC2CN(C(=O)COC3CCC3)CCC12 C1(NC(c2n[nH]c(O)n2)=O)COCCN(C(=O)C2=C(Cl)CC2)C1.C(=O)CSC c1(C(=O)NCCn2cc(C3CCC3)nn2)cccnc1CCOC1CCOC1 CCCC(C(=O)NC(C)CNC(C1CCCCN1C(=O)NC(C)C)=O)OC C(=O)(C1CNC(=O)c2ccnn21)OC.C12CC3(CCC(CC3)C(=O)N1C1CC1)C2 Cc1nc2cc(C(=O)NC3(CO)CCN(C(=O)C=CC4CC4)CC3)ccc2s1 C(=O)(C(F)C(F)(F)F)N1C(C(=O)NCCC(C)(C)O)C=CC1 C(=O)(C1=CCCN(C(c2cc(Br)ccc2C)=O)C1)N(CC=C)CC=C n1(CC(=O)NCC(C)NC(=O)CC2CCC(=O)N2)c(O)nc2ccccc12 c1(C(N(C(CN(C(C2(C(F)F)CC(=C)C2)=O)C)C)C)=O)ncc(Br)cc1F C1(CNC(c2ccc(COC(C)C)o2)=O)C(C2CC2)CCN1C(c1cn[nH]c1)=O Cc1cnccc1C(=O)NCC1CCC1NC(=O)CCOCC1CC1 C1(C(N(CC(C)N(C)C(c2cnc(O)n2C)=O)C)=O)CNC(=O)N1C c1(OC)sccc1C(=O)NC1COCC1C(=O)NCc1ncc(CO)o1 c1(C(=O)NCC(CN(C)C(C2CC(S(C)(=O)=O)C2)=O)O)cc(N)c(N)cc1F N1(C(C(CC#CC)NC(c2coc(CCC)n2)=O)=O)CCn2c(C)cnc2C1 c1(OCC)ncc(C(=O)N(CC(C)NC(=O)C(c2csc(C(F)(F)F)n2)=O)C)s1 C1(C(=O)NC(C(F)(F)F)C2CCCC2)CC2(CCC(F)(F)CC2)C1 C1(C(N(CCN(C(=O)CN(S(C)(=O)=O)C)C)C)=O)CCC1(C)C.C(CO)S CCC(O)CC(=O)NC12CC(C(=O)NC3CCCCC3F)(C1)C2 C#Cc1cccc(C(=O)NCC2CC(=O)N(C)C2=O)c1C N1(C(C=CC)=O)CCC(NC(c2cnn(CCO)c2)=O)C12CCC2 N1(C(CCCC(C)C)=O)CCC2(CC1)CC(C(=O)NCc1ccoc1)CO2 c1(C(N2CCC(CCNC(c3onc(CC)n3)=O)C2)=O)[nH]c(C)c(C)c1C C1(CC)OCCC1C(=O)N(CCNC(c1cnnn1C)=O)CCc1ccccc1 N1(C(c2c(C)scc2)=O)CC2CCCC1C2CNC(=O)C(N1CCN(C)CC1)C c1(C(N2C(CNC(C3(OCC)CCOC3)=O)CC2)=O)cn(C(C)C)c(C)cc1=O C(=O)(C(C)(O)CC)NCC(C)(CNC(=O)CCn1ccccc1=O)OC Cc1ccncc1-c1cn(C2CNC2)nn1.C1CCCN(C(=O)CCCF)C1 C(=O)(C(C)Cc1ccccn1)NCC(C)NC(=O)CSc1nccn1C c1(CN2CC(NC(c3cccc(CO)c3)=O)C(F)C2)cnc2n1CCOC2 c1(C(=O)NC2CC(F)(CNC(CCNC(N)=O)=O)C2)n[nH]c2nccc(Cl)c12 CCC(CCOC)C(=O)N(C(C)C(=O)NCc1coc(C)n1)C1CC1 CCC(CC)C(=O)N(C1CCCC1)CC(=O)NCC(COC)OC N1(C(=O)CC23CCCC2C3)CC2CN(C(C3(C4CC4)CC3)=O)CC2C1 c1(C(=O)NC2CCC(C)(CNC(=O)CC3C=CCC3)CC2)cc(S(N)(=O)=O)co1 C1(C(N2C(CN(C)C(c3cnn(C)n3)=O)CC(F)C2)=O)CC2CCC(C1)S2 CC1NCCN(CC(c2cccnc2)O)C1C c1(C(=O)NCC(CC=C)NC(=O)C(C)(O)C(C)C)ccc2[nH]ccc(=O)c2c1 C1C2CS(=O)(=O)NCC3(CCN1C3)C(=O)O2.C(C)(C)(C)OC.CO c1(C(=O)NCC(O)CNC(C2CCC3(CC2)CC3)=O)cc(O)c(O)c(O)c1 CC(C)C(CCNC(c1c(C2CC2)cnn1C)=O)NC(C1CCCS1)=O C(C)(C(CO)NC(=O)CSc1nncn1C)NC(C=CC(C)(C)SC)=O c1(C(c2nnnn2C2CCOC2)NC2(C=C)CCC2)ncc(Br)cc1OC N1(C(=O)CSC(F)F)CCCC(C(=O)NCC2(N3CCOCC3=O)CC2)C(F)C1 C1(N(C(=O)C=CC2CCCO2)C)CC2CCC(C1)N2C(c1cc(N)cnc1Cl)=O C(=O)(C1=CC2C=CC1C2)N1CC(C(=O)NCCC(CC(C)C)C)N(C)CC1 c1(OC)cccc(NC(=O)CC2CCN(C(=O)CCc3cccc(F)c3)C2)c1C c1(C(C(=O)NCCN(CCOC)C2CC2)OCC2CCC2)ccc(F)cc1 c1(OC)ccc(C(N2CC3CC3(CNC(c3n[nH]c(C)c3F)=O)C2)=O)cc1O Cc1c(C(=O)NCC2CN(C)CCN2C(C2CC3CC3C2)=O)cnc2ncnn12 Cc1noc(C)c1C(C)C(=O)NCC(C)(Cn1cccn1)NC(=O)CNC=O C1(Nc2ccc(C(C)=O)cn2)CN(C(=O)Cc2sc(O)nc2O)CC1(C)C C1(NC(CC(=O)NCC)=O)CN(C(=O)C(C)Cc2ccco2)C2(CCOCC2)C1 c1(C(c2c(C)cc(O)cc2C)=O)[nH]nc2ncc(-c3ccc(F)nc3F)cc12 N12CCCCC1c1n[nH]cc1C2=O.N1(CC2C(=O)NCC2)CC(F)(F)CC1 c1(C2CCN(c3c(C(=O)OC)cncc3)C2)cccc2ccccc12 Cc1cc(=NCC2CNC(=O)C(C)(C)C2)[nH]cc1S(=O)(=O)N(C)CC1CCCS1 c1(C(=O)NCC(CCNC(C2CC2F)=O)OC)cnnc(C)c1 c1(CC)cccc(C)c1C(=O)NCCC1CC(NC(C2CN(C)C(=O)N2)=O)C1 c1(C(N(C2CCCN(C(COCCN(C)C)=O)C2)CCO)=O)cc(=O)n(C)cn1 C1(OCC)COCCC1NC(C1CCN(C(C23CC(C(=O)OC)(C2)C3)=O)C1)=O C(CCC(=O)N(CCCCN(C(=O)C(C)OCC1CCCO1)C)C)NCC=C C(=O)(C(C)C(C)S(C)(=O)=O)N1CC(CNC(c2cnn(CC)n2)=O)OC(C)(C)C1 CCS(=O)(=O)c1ccc(CCC(N2CCC(CN(C(=O)CCF)C)C2)=O)cc1 C1(C(C)C)C(=O)N1.C1(C(=O)OC)(C(=O)NC(C)C2CC2)CC(F)(F)C1 N1(C(c2cnn(C)c2Cl)=O)CCCC(C2(NC(C3C4CCCC34)=O)CC2)C1 C12(OCC)CCC(NC(=O)NC3CC(OC)CC(=O)N3)(CC1)C2 N1(C(CN2CC(C)C2)=O)CCCC2(CCCN2C(c2ccc(F)c(CO)c2)=O)C1 N1(C(CC(=O)NC)=O)CCC2(CC1)CC(NC(=O)CN1CCCCC1)CCO2 C1(C(C)NC(c2cncs2)=O)CCCN(C(c2ccnn2C2CC2)=O)C1 C1(C(N2CC(n3cc(CNC(C4C(COC)C4)=O)nn3)C2)=O)C2CCC(F)(F)C12 CCC(CC)CCC(=O)N1CC2CC2C1CNC(=O)CCC(C)(C)N(C)C CCC(C)(C(=O)N1CCC(C)(CCNC(c2ccc(C(F)(F)F)[nH]2)=O)C1)C(N)=O C1(C(=O)NCc2cncc(C(N(C(C)C)CCF)=O)c2)CCCCC(=O)N1 c1(CC)[nH]nc(C(N2CCC(C(C)(C)NC(c3scnc3Cl)=O)CC2)=O)c1Cl CC12CCC(C(=O)NCc3nccc(C(F)(F)F)n3)(CC1)CO2 C=CCCC(C)(C)NC(c1cnc(CNC(c2ccc(CC#N)cc2)=O)nc1)=O c1(C(=O)NCC2C(C)(C)CCN2C(=O)CC2CC3(CC3)C2)cnc2[nH]ccc2n1 c1(OC)cc(NC(=O)C(C)(CC2CCC2)NC(=O)C(F)C(C)(C)O)ccc1O c1(C(=O)OC)cc(C(N2CC(N(C)C(C3(F)CCOCC3)=O)C2)=O)ccc1OC c1(CC(C)C(N2CCC3C(NC(c4ccnc(S)c4)=O)C23)=O)ccc(F)c(F)c1 N1(C(c2n[nH]c3c2COCC3)=O)CCC2CCN(C(C3(O)COC3)=O)CC2C1 c12nn(C)cc1OC(C)(C)CNC2=O.c1(OC)ncccc1Br Cc1cc(Cl)cc(C)c1NC(c1nnnn1CC1CCOC1)c1cncs1 C12(CCN(C(c3cnn(CC)c3)=O)C1)CCO2.C1(OCC(=O)NC(C)C)CCCOC1 C#CCCCCCC(=O)NCC1CCC2(CN(C(c3ccc(F)o3)=O)C2)O1 C1(C(=O)NC2C(C)N(C(=O)C=CC3CCC3)CCC2)CC2(CCCCC2)C1 CCCCC(CC(=O)N(C)CC1CCOC1)NC(c1cnn2cccc2c1)=O CCCCCCC(CC)C(=O)NC1CC(F)(CNC(c2c(C)nc(C)n2O)=O)C1 C12(CNC(C3(CC)CC3)=O)CCCC(CN1C(=O)CC1CCCCN1C)C2 c1(CSCC)cc(C(=O)N(C)CC2CCCN2C(=O)COC2CCCCC2)no1 C1(C)(C(=O)NCC2(C)N(C(c3nn(C)c(C(F)F)c3)=O)CCC2)CCCCCC1 N1(C(CNS(C)(=O)=O)=O)CCN(C(c2cccc(CO)c2)=O)CC(C)(F)C1 c1(OCC(C)C)cccc(N(CC(=O)N(c2cccc(F)c2)C)C)c1 C1(OC)CCCCC1(C)C.c12ccc(o1)C(c1nnnn1C(C)C)N2.C1(C)(SC)CC1 CN1C(=O)NCC12CN(C(=O)C(c1ccco1)NC(c1cncs1)=O)C2 C1(C(=O)NCCN(C(COCC=C)=O)CC(C)O)CCC(F)(F)CC1 N1(C(C(C)OCC(C)C)=O)CCCC(CC(=O)NC2CCCSC2)C1 c1(C(=O)NCC2C3CN(C(C4CC5(C)OCC4C5)=O)CC32)c(F)cc(F)cc1F c1(OC)cc(OC)c(CC(N2CCC(CN)C2)=O)c(OC)c1 c1(NC(C2CC(CNC(c3cc(C)[nH]c3C)=O)C2)=O)ccc2n[nH]cc2c1 CCC(F)(F)C(=O)N1CC(NC(c2ccc(COC)nc2)=O)C(C)C1 c1(CNC(c2ccc(C(C)=O)[nH]2)=O)nc(C)c(C(=O)NCCc2cocn2)o1 C(=O)(C1=C(C)CCCC1(C)C)N(C(C)CNC(=O)Cc1sc(C)nc1C)CC N1(C(c2ccc(Cl)cc2)C2(N)CC2C(F)(F)F)CCCc2[nH]ccc2C1 c1(C(=O)NCCC(C(C)C)NC(CC2(C=C)CC2)=O)c[nH]c2nccc-2c1 c1(C(=O)NCCCCc2cn(Cc3csc(Br)n3)nn2)ccc2c(c1)CCC2 N1(C(c2c(OC)cccc2)=O)CCCCCC1CNC(c1ccc(C)cc1O)=O C12(CNC(CC3C(C)CCO3)=O)CCC(CC1)N(C(C1(C(F)F)CCCO1)=O)C2 C1(C(=O)NCC#CCNC(Cc2nnc(C)n2C)=O)CC12CC(F)(F)C2 C(=O)(C(CNC(C1CC1F)=O)CC(C)C)NCc1c(C)cc(C)nc1 C1(O)(CCNC(=O)Cc2ccon2)CCN(C(=O)CCN2CCOC2=O)C1 c1(OCC)nccc(C(N2CCC(C(C)NC(c3cnccc3C)=O)C2)=O)c1F c1(C(N2C(C(C)NC(=O)CCC(N)=O)CCCC2)=O)cccc2c1CCC2 C(=O)(CCC#Cc1ccccc1)N(C1CN(C(=O)C(F)(F)c2cncs2)C1)CC C12(C(=O)NCCC(COC)(C)C)COC(C1)C(NC(=O)C1CC1)C2 N1(C(C2(C)CCC2)=O)CCC(C)(C)C(CNC(=O)COC(F)F)C1 Cc1ccc2c(C(=O)NCCc3ocnc3CNC(=O)C=C3CCC3)c[nH]c2c1 c1(C(N2CC(O)(CN(C(C3C(C)C3C)=O)C)C2)=O)coc2c1COC2 c1(SC)nc2ncnc(N3CC4CC(NC(C5(C)CC6CCC5C6)=O)C4C3)c2s1 N1(C(C(C(C)C)N(C)C)=O)C(CC(=O)NCCC(C)N(C)C)C2CCCC12 C1(C(NOCC(=O)NCC)=O)(CNC(=O)C(C)CO)CC(C)(C)C1 N1(C(C(C)n2cccn2)=O)CCS(=O)(=O)C(CCNC(C2(O)CCSCC2)=O)C1 Cc1cc(F)c(Cl)cc1C(=O)NC1CC(CNC(=O)C2=CCC2)C1 n1(CC)nnc(C)c1C(=O)NC(C1CCCCC1)CNC(C1CCS(=O)(=O)C1)=O C1(NC(c2coc(Cl)n2)=O)CN(C(C2CC(=C3CC3)C2)=O)C2CC12 C1(C(N(CCC)CCN(C)C)=O)CCCN(C(=O)C(C#N)C(C)C)CC1 C(=O)(N=c1cc[nH]cc1Cl)c1cccc(CNC(=O)Cc2cscn2)c1 c1(C(=O)OC)cccc(C(O)COC)n1.c1(CNS(=O)(=O)CC2CCC2)ccccc1 c1(C(=O)NC(C)CCCNC(=O)COC2CCCCCC2)cccc(F)c1C#N CC1(C)C(C)(C(=O)NCC2CCCC2NC(C2(C3CC3)CC2)=O)C1(C)C c1(NC(C(=O)NC(c2c(F)cccc2F)CC(C)C)=O)c(Cl)nc2ccccn12 c1(C(=O)NCC(C)(Cn2cccn2)NC(=O)CCOC2CC2)ccc[n+]([O-])c1 CCC1CCCC(=O)N1.C(C)(C)(C)OC(=O)NCCN(C(C)C)C(C)C C1(C2CCC2)(C(N(C(CNC(c2c(C)coc2C(C)C)=O)C2CC2)C)=O)CCC1 N12CCN1CC2CO.c1(C=O)c(C2CC2)cccc1F.C=CCCCC=O C1(NC(=O)CC(F)F)CC(NC(=O)Cc2cccnc2F)C(O)C1 N1(C(Cc2ccc(C)nc2Cl)=O)CCC2(C1)CN(C(c1ccc[nH]1)=O)CC(C)O2 c1(C(=O)NCC2(CC(N3CCC(OCC=C)C3)=O)CC2)ccc(=N)[nH]n1 CC1(C)CN(C(=O)C(=O)NCC(F)F)CC1NCCCN1C(=O)CNC1=O c1(C(=O)NC2CC(NC(C3(N(C)C)CCC3)=O)C23CCC3)c[nH]c2ccncc12 C1(=CC(=O)NC(CN(C)C(c2cc(C(F)F)cs2)=O)(C)C)CC2CCC(C1)N2C N1(C(c2c(NCC)scn2)=O)CCOCC(CNC(=O)CC(C)CF)C1 N1(C(C=C(C)C(F)F)=O)CCN(C(c2cnn(CC3CCCC3)c2)=O)C2CC12 c1(NC(C(C(C)C)=O)=O)ccc2c(c1)CN(c1ncc3ccccc3n1)C2 N1(C(C2(C)CC=CC2)=O)CC2CCC2(C(=O)NCCc2ccoc2)C1 Cc1nn(C)cc1CCC(=O)NC1CC1CNC(=O)Cc1nc[nH]n1 Cc1[nH]c(-c2nc(-c3ccc(Cl)c(COC(C)C)c3)nn2CF)c(C)c1C(C)C C1(NC(=O)CNC(C2C=CCN2C(c2ccnc(S)c2)=O)=O)CCCC(F)(F)C1 Cc1ccc(Cl)c(C(=O)NCC2CC3CCC2N3C(c2ccc(C#N)s2)=O)c1 c1(C(N2CCN(C(CC(CC)SC)=O)CC2C(F)F)=O)ccc2c(ccn2C)c1 C(C)(C(=O)NCC1CCCN1C(c1cnc(C)[nH]1)=O)(C(C)C)NC(C)=O C(C)(CNC(c1cccnc1N)=O)(CC(C)C)NC(c1cc(SC)c(C)o1)=O N1(Cc2cc(C)no2)CCC(O)CC1C(=O)NC(c1ccccc1Cl)C c1(C(N(C(CCSC)C)C)=O)cc(Br)c(F)cc1Cl C(CCCC(CO)NC(=O)CSc1nncn1C1CC1)NC(COCC)=O c12ccc(cc1)OC(=O)C2.C(C(C)C)N(C(C)C1CC1)CC O=C(CC1=CCCCC1)NC1CCCC2CN(C(C3CC(C(F)(F)F)C3)=O)CC12 N1(C(c2c(CC)nns2)=O)CC(NC(C2CN(C(C)C)CCO2)=O)CC1(C)C N1(C(c2c(C)ncn2O)=O)CCN(C(=O)C(C)Sc2ccccn2)CC(C)(C)C1 Cc1n[nH]c(C)c1CC(C)C(=O)NCC1COCCN1C(=O)COc1ccsn1 CCCC(C(=O)NCC(c1ccccc1)NC(c1cncc(C2CC2)c1)=O)OC c1(OC)ccc(C(=O)NCCOCCN(C)CCN2CCCCC2)c(C)c1 N1(CCC)CCCC1C(=O)NC1CCC(NC(=O)COCCSC)C1 C1(CC(=O)NC2CCCC2NC(C2CCCCO2)=O)CCCC1(F)F c1(NCCOCC(C)C2CC2)ccc(S(=O)(=O)NCC2CC=CCC2)cc1Cl Cc1c(Cl)sc(Cl)c1C(=O)NCCC(C)NC(c1c(F)cccc1F)=O N1(C(c2ccsc2)=O)CCOC2(CCN(C(c3nc(Cl)sc3Cl)=O)C2)C1 C1(NC(c2n[nH]c3c2COC3)=O)CCCN(C(=O)CC2CCS(=O)(=O)CC2)CC1 CC1(C)CN(C(C2(C#N)CCCO2)=O)CCC1NC(=O)CCCc1ccccn1 c1(C(=O)NCC2CCN(Cc3cccc4c[nH]nc34)C2)ccc(Cl)cc1[N+](=O)[O-] Cc1cc(N)c(C(=O)OCc2cccc(C(C)(C)F)c2)cc1C C(CCC(=O)N(CC(C)O)CCNC(=O)C(F)=C1CCC1)SC CC1(C(=O)NC(CO)C2CCC2)CC(NC(c2cn(C3CC3)cn2)=O)C1 C(CCCCC(=O)N1CCN(C(=O)COCC(F)F)CC1CCO)OC(C)=O c1(C(=O)NC(C)CCCNC(=O)Cc2ccco2)coc2cc(F)ccc12 C1(NC(C2CC(SC)C2)=O)CCCC(NC(c2ccc(SCC3CC3)cn2)=O)C1 C(=O)(C1=CCCOC1)NCCC1CCC(NC(=O)CNC(N2CCCCC2)=O)C1 C1(C(=O)NC2CCOC2C(N2CCCC(C(C)(C)O)C2)=O)(CC)CCCCO1 CCCC(C)CC(=O)NCC(C(N1CC2(CO)CCC1C2)=O)N(C)C C1(C(=O)NCc2cc(C)sc2)CCCCN1C(c1cc(C(N)=O)[nH]n1)=O N1(C(c2occ(C)c2)=O)C(C)CC2CN(C(=O)CCC3CCC(=O)N3)CC12 Cc1c(C(N2CCC3(CC3C(=O)N(C)OCc3ccccc3)C2)=O)cccc1Cl Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(=O)C(O)CN2CCCC2)C1 c1(C(=O)NCC(n2cc(C3(N(C)C)COC3)nn2)C)ccccc1C(C)(C)C#N c1(Oc2cccc(C3(C)CC3)c2)cccc2ccccc12 [N-]=[N+]=NCC(C(=O)NCC1CC1Cl)NC(=O)Cn1cnc(=N)[nH]1 c1(C(N2CC(NC(C(C)O)=O)C(F)CC2)=O)cccc(P(C)(C)=O)n1 C1(C(=O)NCC(COCC)C)C2CC(O)C(C2)N1C(C1(C(C)=O)CC1)=O C1(C(=O)NCc2c(C(=O)NCc3cnc(C)s3)occ2)CCC(O)CN1C c1(C(=O)NC2CCN(C(c3[nH]cc(CC)c3)=O)CC2C)cccc2cc[nH]c12 C1(NC(C2CCC(CC)O2)=O)CCC12CCN(C(c1cc(C#N)c[nH]1)=O)CC2 Cc1cc(C(=O)NCCC2CCN(C(=O)Cc3cnccc3Cl)C2)nn1C CCC(CCNC(C)=O)C(=O)NC.C1(=O)CNC(=O)N(C)CCN1.C(CO)N c1(OCC(=O)N(C(CC(=O)NC(CC)C)C)C)ccc(C(=O)NCCCO)cc1 N1(C(CN(C)C)=O)CCC(n2ccc(NC(=O)Cn3cncn3)n2)CC1 N#Cc1ccc(C(N2CCC(NC(c3nc4c(s3)COCC4)=O)C2)=O)c(F)c1F N1(C(=O)NCc2ccc(F)c(C(F)(F)F)c2)CCc2cc(OC(F)F)ccc2C1 N1(C(Cn2cc(C(=C)C)nn2)=O)CCN(C(=O)NCc2ccccc2)CC12CCC2 C(=O)(C(CCOC)NC(=O)C(Cl)Cl)NCCC(C)N(CCC)C C1(CNC(CC2(OC)CCC2)=O)CN(C(c2cncn2C)=O)C2CCCC2O1 Cc1ccccc1C(C1CCCC1)NC(=O)C(C(C)C)NC(=O)C(C)(C)O c1(C(=O)NC2C3N(C(C4(CC=C)CC4)=O)CC(CC3)C2)cc2cccc(F)c2o1 C1(Cn2c(N3C(C)(C)CCC3)nnc2C2CCCCO2)CC2(CCCC2)C1 CC(C)CC(N=c1[nH]c(=NC2CC(F)(F)C2)[nH]c2c1COCC2)c1ccc(Cl)s1 c1(OC)ccc(-n2nc(-c3nc(C)cs3)nc2C2CN3CCN2CC3)c(C)c1 C1(C(=O)NC(c2cn(C)nn2)C(=O)NCC2(C#C)CCC2)(CO)CC=CCC1 C1(OC)C(NC(=O)N(Cc2ccc(F)cc2)Cc2ccccc2F)C2CCCC12 c1(CC(=O)NCCCNC(C(C)c2ccon2)=O)ccc(Cl)cc1Cl N1(C(C)=O)CCCC(C(N2CCCC2CNC(=O)CCc2csc(=N)[nH]2)=O)C1 C12(CNC(C(CC)CC)=O)CCC(CN(C(c3n[nH]c4c3CCSC4)=O)C1)C2 c1(NC(=O)NCC2CCN(C(F)F)C2)ncnc(C(F)F)c1Br Nc1ccc(F)c(F)c1C(=O)NCC1CC1NC(C1CC(=O)NC(=O)C1)=O Cc1ccc2oc(C(N3CCn4cccc4C3C)=O)cc2n1 CC1CN(C(=O)C(=O)NC2CCC(=O)C2)CC2(CCN(C)C2=O)C1 C12(C(N(CC(C)OC)C)=O)CC(CCO1)N(C(=O)C(C)C1CCCO1)C2 n1(CC(=O)NC(CNC(c2csc(C)c2C)=O)(C)C2CCC2)nc(O)ccc1=O N1(C(CCC=CC)=O)CCCC2C1CCCCN2C(=O)C(N1CCCC(C)C1)=O c1(C(C(=O)NCCC(=C)CNC(c2ncccc2F)=O)F)cccc(C)c1 C12CN(C(C)(C)C1)C(=O)CN2.Cc1c[nH]nc1CNC(=O)C1CC1 N1(C(C2(O)CCN(C(C3CCN(C)C3)=O)C2)=O)CCc2ccsc2CC1 N1(C(c2c(CCC)nco2)=O)CCC(CF)(NC(C2CC3CCC2O3)=O)C1 N1(C(c2c(CCOC)occ2)=O)CCN(C(=O)CNC(=O)C(C2CC2)SC)CC1 c1(N2CC(OC)C3(C2)CC3)ncc(C)cc1S(=O)(=O)NC1C=CCCCC1 C(C1=CCCCC1)(c1n(CCCSC)nnn1)NCC1CC=CCC1C Cc1coc(C=CC(=O)NCC(C2CC2)NC(=O)Cn2cc(C3CC3)cn2)n1 c1(C(=O)OC)cncc(-c2cn(C(C)C(N3CC(O)CC3C)=O)nn2)c1 N1(C(C2C(C)CCC2)=O)CCC2(CC1)CN(Cc1ccc(F)c(O)c1)CCO2 C(CN=c1[nH]cncc1I)(C(C)(C)C)NC(c1ccn(CCOC)n1)=O C1(NC(c2c(COC)ncs2)=O)CC(F)CN(C(c2cnoc2C)=O)C1 N1(C(CC(C)(C)C)=O)CCC2CCC(C1)N2C(=O)C(F)(F)C=Cc1ccccc1 C(=O)(C(C)P(C)(C)=O)N(C(C)C)CCNC(=O)CC1CCNC(=O)C1 N1(C(c2c(CC)n(CC)nn2)=O)CCOc2cc(C(C)(C)C)ccc2C1 C1(C(=O)NC2C(NC(=O)CCC3CCCC3)COCC2)CCC(F)(F)CO1 C1(NC(C(C)C)=O)CN(C(c2nccnc2N)=O)CC1(C)C c1(CNC(C2CCN(c3ncccn3)C2)=O)ccncc1Cl c1(CC)cc(F)cc(F)c1.C12(C(N3CCCC(OC)C3)=O)CCN(CC1)C2=O CC1NC(=O)C2=C1N(c1ccccc1)C(=O)NC2c1c(C(=O)O)cnn1CCO c1(C(C)C)ccc(C(=O)NC(C2CCOC2)CNC(C2CCOC2=O)=O)s1 C1(C2(NC(=O)CCNC(c3cc(C)c(C)s3)=O)CC2)(OC)CCC1 C1(C(=O)NC(CC=C)(C)C)CN(C(=O)CSC)CC1C CC12CCOC(CNC(c3cc(OCC(F)(F)F)c(Cl)cn3)=O)(C1)C2 Cc1cnc(C(=O)NCc2ccc(CNC(C3(C)CCNC3=O)=O)cc2)cc1Cl C=C(Cl)CC(C(=O)N1CCC(O)C(C)C1)NC(=O)CC N1(C(C(CC)C#N)=O)C2C(CO)CC1(C(N1CCOC(C)(C)C1)=O)C2 C=C1CC(C(=O)NC2CCCC2C)(CNC(=O)CCN(C2CC2)CC)C1 C1(CNC(Cc2c(C)cco2)=O)CC(NC(=O)C(C(C)C)n2cccc2)CCO1 CCC(C(=O)NCC(C)(C)OCC(=O)NCCC(C)C(C)(C)C)C(C)(C)CC C(=O)(C1=CCCCC1)NC(C(=O)NC1(C)CCNC1=O)CCNS(=O)(=O)C1CC1 C=C=CCC(C(=O)OC)NC(=O)CCC1(C)CCC1.c12ccc(cc1)c(=O)[nH]2 C(=O)(CCCCC(=O)NCC(C)(C)CCNC(c1nccc(Cl)c1F)=O)OC C(CCC)(C(=O)NC12CC(C1)N(C(=O)C(C)N(C)Cc1ccccc1)C2)=CCC C12(C(N3CC=C(CNC(CCc4ccc(C)s4)=O)CC3)=O)CCCCC1C2(F)F C1(NC(CCN2CCN(C)CC2)=O)CCCN(C(C2CCCC(F)(F)C2)=O)CC1 c1(NCC2(F)CN(C(C3(C(=O)OCC)CC3)=O)C2)cc(=O)n(C)cn1 Cc1cc(C(=O)NC2CC3CC2N(C(c2ncc(C(F)F)s2)=O)C3)cc(C)c1F N1(C(C(=O)NCC)=O)CC(NC(=O)CCOCC(=O)OCC)CC(F)(F)C1 c1(-n2c(C3C(CF)CCC3)nc(C3CCCC3)n2)cccc2cnccc12 C1(OC)CC2CC1CN(C(=O)C(CNC(C1CCC(=O)N(C3CC3)C1)=O)C(C)C)C2 C(=O)(C(C(C)(C)C)NC(c1ncccn1)=O)N1C(C)(CC(=O)N(C)C)CC1 c1(C(=O)NC(C(c2ccccc2)NC(CCC2C(C)C2)=O)C)cc(C#N)no1 C=CCC(C)C(=O)N1CC=CC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1 C(C(C1CC1)(C1CC1)OC(C)(C)C)(OC)NC(=O)NCCNCC1CCC1 C(=O)(C1=CCCS1)N(CCCNC(=O)C(F)(F)C1CCCC1)CCC c1(CNC(C2(CNC(C(N3CC(C)C3)C)=O)CCCC2)=O)cccc(F)c1F C1(C(N2CCCC(OCC)C2)=O)CN(C(c2cc(C)oc2C)=O)CC(C)(C)C1 CCCCC(C(=O)NCC(CNC(c1cc(CO)sc1)=O)OC)NC(N)=O c1(CNC(CN(CCC)C(c2c[nH]nc2Cl)=O)=O)nocc1CC C1(C(=O)NC2CCN(C(C3CC(C)(C(=O)OC)C3)=O)C2C)CCC2(CCC2)O1 N1(C(=O)NCC(C2CCCCC2)C)CCOCCC12CCOCC2 C1(CNC(C=CCCC)=O)CCN(C(c2nc(OC)ccc2F)=O)C(C)C1 N1(C(CSCCCC)=O)CC(NC(c2csc(C(N)=O)n2)=O)CC(C)C1 c1(C(N2CCC(O)(C(C)NC(=O)CS(C)(=O)=O)C2)=O)cn(C)c(=O)nc1O C(c1ccc(C2CC2)cc1)=CC(=O)NC(C(CO)NC(C=CCOC)=O)C C1(COC)(CNC(=O)C(C)OC2CC2)CCCN1C(c1coc(SC)c1)=O C(=O)(C(F)(F)CC(C)C)NC(CC(C)C)CNC(=O)CC(C)N1CCCC1=O C1(C(NOCCCC(=O)OC)=O)CCCCCN1C(C1CCC1C)=O n1(CC)ccc(C(=O)NC(C)CCN(C(=O)Cc2nc(C(F)F)nn2C)C)c1C CN1CCOc2cc(NC(=O)CC3COCCN3C(C3CC3(C)C)=O)ccc21 N1(C(c2ccc(CC)cc2)=O)CCN(C(c2[nH]ncc2C)=O)CC1CC(=O)NC c1(C(=O)NC(COC)CNC(C2C=CCC2)=O)ccncc1 c1(C(=O)NC(C)CO)nn2ccccc2c1C(=O)NCC1CCOC1 c1(CC(=O)NC(CC)CN(C(=O)CCOC(C)C)CC)ccc(O)cn1 C1(C(=O)NC2(C(=O)OCC)CC2)CN(C(C2CC3C=CC2CC3)=O)C2(CCC2)C1 CCCCC(C)C(=O)N1CC(F)CC1CNC(C1CCS(=O)CC1)=O C1(C(=O)NC(C=CC(=O)N(CC(C)C#N)CC)C)CC1C1CCC1 Cc1nc2ccc(C(N3CCC(F)C(NC(=O)CCC4CC4(F)F)C3)=O)cn2n1 C(=O)(CCCCCF)N1CCC(C)(NC(CCCOc2ccc(C)cc2)=O)C1 N1(C(Cc2cnc(C)[nH]2)=O)CCN(C(=O)CCSCC(N)=O)C(CC(=O)NC)C1 c1(C(N(CC(=O)NC)C)=O)ccc(CNCCNS(C)(=O)=O)cc1 C#CCC(CC(=O)N1CCCCC1C(C)(C)C)NC(=O)CC(C1CC1)C1CC1 C1(CNC(c2sccc2F)=O)CN(C(=O)CC2CC=CCC2)CC1C(F)(F)F C(C(C)(CO)CN=c1cc(C)c(S(=O)(=O)Nc2cncc(C)c2)c[nH]1)OC Cc1ccc(C(O)C(=O)NC2CC(NC(C3CCNC(=O)C3)=O)C2)cc1 C(=O)(C(C)(C)CO)NC1C(NC(C(n2ccc(C(F)(F)F)n2)C)=O)C1 CCC(C)CC(=O)N1CCC(C)C1CNC(C1(COC)C=CCC1)=O C(=O)(C#CC1CCOC1)NCCCCNC(C(c1ccc(C#N)cc1)O)=O Cc1nc(SC(C)(C)C)nc2c1NC(=O)C(C)N2C C1(CNC(c2c[nH]c3ncccc23)=O)CC2CCC1N(C(=O)C1=CCC1)C2 O=C(CN=c1nc[nH]s1)NCC(C1CCCC1)NC(C12CCOC1CCOC2)=O c1(OC)cccc(CCC(=O)NC2CC(C)(NC(=O)C(F)C3CCOC3)C2)c1 CC(C)(CC(F)(F)F)C(=O)NCC1CCCN1C(C1(CCN(C)C)CCCC1)=O c1(OC(COC)CNC(c2cc(Cl)sc2C)C(=O)OC)ccccc1C C(CC(O)C(=O)NCC1CCC1NC(=O)C(F)(F)CC1CCCO1)N(C)C c1(C(N(C(CCNC(C(C)c2cccs2)=O)C)C)=O)c[nH]c(=O)cn1 C1(CC)CCN(C(c2scnc2Br)C(=O)NCc2ccc(Br)cc2)C1C N1(C(C2(OC)CCCOC2)=O)CC2(C1)CN(C(=O)CCCCO)CC(C)(C)O2 CCC(C)(CO)C(=O)NCC1CC(F)CN1C(C1CCC(=O)N1C1CC1)=O C(CCC(N)C(=O)NCCSCc1ccc(Cl)c(Cl)c1)OC [N-]=[N+]=NCCCC(=O)NC1CCCCC1NC(c1ccccc1CC#N)=O CC1=C(C(=O)N2CC3CCC2C(CNC(=O)CCc2nc(O)n[nH]2)C3)SCCO1 c1(SC)nc(N2CCCC(C)(C(N3CCC4(CC3)COC4)=O)C2)ncc1F N1(C(c2n(CC)ccc2)=O)CCC(NC(=O)CC(C)(O)COC)C(F)(F)CC1 C(=O)(C1c2c[nH]nc2CCC1C)NC1CCCCN(C(CCC(C)O)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)C=CCC)N1CCCC(CCC=C)C1 c1(OCC)nc(N2CCC(NC(c3cc(C(F)(F)F)cs3)=O)C2C)ncc1Cl C12(NC(C(CCOC)OC)=O)CCCC1N(C(c1cc(C)nnc1O)=O)CCC2 c1([SH](N2CC(NC(=O)NC(=O)C(=O)C3CCCC3)C2)C)ccc(-c2ccccc2)[nH]1 C1(C(=O)NCC2N(C(c3cn(CC)nc3)=O)CCC2)CC(=O)NC1(C)C C1(C2CCN(C(C3COCCC3C)=O)CC2)(NC(c2[nH]c(=NCC)sc2)=O)CC1 N(C1COc2ccc(F)cc21)C(CN1CCN(C(Cc2cc(C)nn2C)=O)CC1)=O c1(CC)ncc(C(C(=O)NCCCC2CC2)N(C)CC2(C)CCCO2)[nH]1 Cc1cc(-n2nc(CCC(C)C)nc2-c2cc(C3CC3)[nH]n2)cc(C)c1 CC1(C)CN(C(C2Cc3ccccc3O2)=O)CC(CNC(=O)C=CCN(C)C)O1 C12(C(=O)OCC)CC3CC(C1)CC(C(=O)O)(C3)C2.C12COC3CN(CC13)OC2=O C1(C(N(C2(C(=O)NCC3(CO)CC3(C)C)CC2)C)=O)CC12CCOCC2 c1(C(=O)NC(C(C)C)CO)ccc2c(c1)CN(C(c1cnccc1Br)=O)CC2 C1(NC(CN(C)CC)=O)CCOC(C(=O)NCC23CC(OC(C)C)(C2)C3)C1 C1(C(=O)NC2CCCC2CN(C)C(C23CCC(CC2)C3)=O)(OC)CCSCC1 N1(C(c2ccc(C(=O)OC)n2C)=O)CCN(C(=O)C(F)C(C)C)C(C)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(NC(c2ccnc(O)c2F)=O)C(C2CC2)C1 N1(C(=O)OC(C)(C)C)C2CCC1(CNC(=O)C(=O)C1CCC1)CC2 C1(OC)CCCN(C(=O)C(Cn2cccn2)NC(=O)C(c2ccn(C)c2)C)CC1 N(C(=NCCC(O)C(F)(F)F)N1CCC(C(F)F)C1)CCC1CCS(=O)(=O)C1 c1(COC)nc(NCC2CCC(C)CC2)cc(=NC2CCC=CCC2)[nH]1 N1(C(C(C(C)C)SC)=O)CCN(C(c2ncoc2C2CC2)=O)CC1C(C)(C)C N1(C(C2CCN(C(=O)NC)CC2)=O)CC(C2(NC(C3COC(=O)O3)=O)CC2)C1 C1(OCC)CCC1C(=O)N(CC(O)CF)C N1(CC(C2C=CCCC2)=O)CCN(C(=O)Nc2cccnc2)CC1 c1(C(N(C2CN(C(=O)CCc3nncs3)CC2F)C)=O)cccc2nsnc12 Cc1cc(O)ccc1C(=O)NC1CC(C(F)C(=O)Nc2cncc(C3CC3)c2)C1 N1(C(C(CC)=CC)=O)CCC(C(=O)NCCc2cc(CC)no2)(OC)C1 C12(C(=O)NC3C(OC)CN(C(C4CC(N(C)C)C4)=O)C3)CCC(C(F)F)(CC1)C2 c1(C(N(CC(=O)O)C)=O)cccc(-n2cc(C3CCCCO3)nn2)c1 C=CCCCC(C(=O)NC1CC2(CCC2)C1OC)NC(c1ccc(O)cc1)=O C1(C)(NC(c2c(C)cno2)=O)CCCN(Cc2ccc(Cl)c(F)c2)C1 N1(C(C(F)=C(C)C)=O)CC(C(=O)N(CCCCO)C(C)C)C(C2CC2)C1 C1(CNC(C(CO)N(C)C)=O)COCCN1C(=O)CC1CCCCN1C C1(N(C(Cc2cnc(C)s2)=O)C)CCCN(C(C2(C)CCOC2)=O)C1 C1(C(N(CCF)CC)=O)CC12CCN(C(C1CCOC1C)=O)CC2 c1(CC)nocc1C(=O)NCCN(CC(C)O)C(c1nnc(C(C)(C)C)s1)=O c1(C(N2CCC(CCNC(C(CCC=C)(C)C)=O)C2)=O)cc2ccc(Cl)cc2[nH]1 CC(CN(C)C)CCC(=O)NC(CN(C)C)C(=O)N(C1CCCC1)CCO c1(C2C(C(=O)NCC(CNC(C3(CSC)CC3)=O)O)C2)cccc(O)c1 c12cccc(c1)C(=O)OC2.CC(C)(C(F)(F)F)c1cccc(NCCO)c1 CCC(C)CCC(=O)N1CC(NC(=O)Cn2cnc([N+](=O)[O-])n2)CCC1C N1(C(C(n2cc(CCC(CC)O)nn2)C)=O)CCc2nnc(C(=O)O)cc2C1 n1(C(C)C)ncc(C(=O)NCC(C2CC2)NC(C2(CO)COC2)=O)n1 C1(C(N2CCC(NC(CCOCC)=O)(CF)C2)=O)CC(c2ccccc2F)=NO1 c1(NC(CNC(C)=O)=O)cc(S(=O)(=O)NCC(CO)NC(=O)C(C)C)ccc1C Cc1cc(Br)c(F)cc1CNC(C1CCN1C(c1cncn1C1CC1)=O)=O N1(C(COc2c(OCC)cc(F)cc2)=O)CCn2ncc(O)c2C1 c1(C(N2C(CNC(c3c(CC)ocn3)=O)CC2)=O)cc2nc(C)sc2[nH]1 c1(C2(C(=O)NC(C)CCN(C(=O)C(C)(F)F)C)CCC2)cccc(Cl)c1Cl N1(c2n(CC=C)c(-c3ccccc3OC)nn2)CCC(C2CC(O)C2)CC1 c1(C(N2CCC(NC(c3c(F)cccc3F)=O)C(O)C2)=O)cc2cccn2cn1 CN(C)S(=O)(=O)NCC(N1CCC(N2CCN(C(C3CC3(Cl)Cl)=O)CC2)CC1)=O c1(C(=O)OC)ccc(CN(C)CC2CCN(C(=O)OC(C)(C)C)C2)cc1 C1(NC(c2ccc(O)cc2C(F)(F)F)=O)CCCCN(C(=O)Cc2ccsn2)C1 c1(COC)nc(NCC2(COC)CCCCC2)cc(=NCc2nn(C)cc2Br)[nH]1 C(CC(C)(C)C)(C(=O)NCCCN(C1CCCC1)C(C1CCC(=O)N1)=O)OC C1(CNC(CSCC=C)=O)(COC)CCCN1C(=O)CCc1cccc(C)c1 C1(CCC)CCCN(C(=O)C(CNC(C2CC3(C2)CC3(F)F)=O)N(C)C)CC1 N1(C(C2C(C)(C)C2)=O)CC2CCN(C(=O)C=CCO)CC12.C(=O)(C(F)(F)F)N c1(C(=O)NC2C(NC(CCC(=O)NCCC)=O)C2)ccc2c(c1)C(C)CN2 N1(C(C2N(C(CN=[N+]=[N-])=O)CC(O)C2)=O)CC2(CCOC(=O)N2)C1 c1(C(N(C2C(C)CCN(C(C=CCC)=O)C2)C)=O)ccc(S(=O)(=O)NC)cn1 c1(CC(C)C(=O)N2CCC(OCCCO)C2)ccccc1F c1(C(N2CCC(O)(CNC(C3CC(CF)C3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] C1(=CCNC(C2C(CC)OCC2)=O)CCN(C(=O)CC23CCCC2C3)CC1 N1(C(COCCC(C)C)=O)CC(F)CC1CN(C)C(c1ccc(OC2CC2)cc1)=O CC1(C)CN(C(C2CCS(=O)(=O)C2)=O)CCC1NC(C1CCCCC1)=O C1(NC(C(C)OC)=O)CC(F)CN(C(c2ccc(I)cc2N)=O)C1 CC(CC(=O)NCC1C2CN(c3ncnc4cnn(C)c34)CC12)CC(C)(C)C C12(NC(C3CC4CCC3O4)=O)CCCC1N(C(c1ccoc1Br)=O)CC2 Cc1cc(F)ncc1NC(C1COCCN(C(C2(N(C)C)CC2)=O)C1)=O c1(C(=O)NC(CC=C)CNC(C2CCC(O)C2)=O)cccc(C(N)=O)c1F N1(C(c2ccc(OC)o2)=O)CC=C(CC(=O)N2CC(N(C)C)C2)CC1 c1(C(=O)NCC(C)CN(C(=O)CC(C)(C)C)C)cc(Cl)c(F)cc1[N+](=O)[O-] C1(NC(C2C(C)(C)CC2)=O)CCN(C(c2ccc(O)nc2)=O)CCC1CO C(CCN)(C(=O)N(C)OC)N.C(=O)(C(C)(C)C)C(C=C(C)C(C)C)=O c1(NC(CCC)C2CC2(C)C)nc(C)cc(=NCC#CC)[nH]1 n1(C(C2CCC2)CN)nnnc1C(C)(CC1CCC1)OC.C(CCO)CC(C)(C)C C(=O)(CCC(=O)C1CC1)NC1C(C(N(C2CCOC2)CC)=O)CC1 n1(C(C)C)ccc(CC(N2CC(N(C)C(C3CC=CC3)=O)C2)=O)n1 C1(CNC(c2ccc(CNC(c3ccc(Cl)o3)=O)o2)=O)(CO)CC2CC2C1 C12(NC(C3C(C(=O)OCC)C3)=O)CCCC(NC(=O)CC3CCCCO3)(C1)C2 c1(NC(CC(C)N(C(CC(C)F)=O)C)=O)cnc(Cl)nc1 N1(C(=O)NC)CC(C)CN(C(=O)NCCNC(=O)OCC)CC1C CCC(C(=O)N1CC(F)(CNC(=O)C#CCN(C)C)C1)n1ccc(C2CC2)n1 C(CCCCCN(C(=O)Cn1cnnc1O)C)NC(COCCCC(C)C)=O C#CCCCC(=O)NCC1C2CN(C(=O)C(O)CCC)CC12 n1(CCC(N2CCC(CN(C(=O)CC3CC3)C)C2)=O)c(=O)n(C)c2ccccc12 c12coc(n1)C(N1CCC1)C(=O)N2.C1(C(=O)OC)(SCC)CC1(F)F.C(C)SC.CC c1(-c2cn(CC(C(C)C)NC(c3ccc(F)nc3)=O)nn2)ccc(F)cc1Cl C(CNC(c1cc(C(F)F)no1)=O)(CC(F)(F)F)NC(C1CCC(=O)C1)=O C(=O)(C1=NOC(C)(C)C1)N(C(C(=O)N(c1ccccc1)CC)CC(C)C)C Cc1ccc(CN2CCCC(C(=O)NCCC3CC3)C2)cc1Cl c1(C(=O)NC(CNC(C2CC(C(C)=O)C2(C)C)=O)C)ncc2[nH]ncc2n1 CC1(CNC(c2ccncc2F)=O)CCCN(C(=O)C=CC=C(Cl)Cl)C1 N1(C(C(n2ccc(C)n2)C)=O)CCN(C(=O)CN2CC3CC3C2)C(CO)C1 CC(CN(C)C(C1CCCC12CCOCC2)=O)N=c1[nH]c2cc(Cl)cc(Cl)c2o1 C1(CNC(c2nc(COCC)sc2)=O)CCN(C(c2cc[nH]c2C)=O)CC1C c1(CC)oc(C)cc1C(=O)NC1CC(NC(=O)OC)C1.C12C=CC(C1)CC(=O)N2 C1(CC(N2CCC(NC(C3N(CCC)CCCC3)=O)CC2)=O)CCCC(C)(C)C1 N1(C(C(C)N(CC)CC)=O)CC2CC1C2NC(=O)C=CCCc1ccccc1 Cc1cc(C(=O)NCC2CCC(F)(CNC(=O)C(C)CC3CCC3)C2)ccn1 N1(Cc2nnc(CC)s2)CCC(NC(c2csc(-c3ccco3)n2)=O)C(O)C1 N1(C(c2noc(CC)c2C)=O)CC(C)CN(c2ncc(C(C)(C)O)cn2)C(C)C1 C1(O)(CNC(C(C#C)(C)C)=O)CCCN(C(c2ccc(N)cc2C)=O)CC1 c1(CC(N2C3CC(NC(CSC)=O)C2CC3)=O)nc2ccccc2[nH]1 C(=O)(CCCCN1CCOCC1)NCC1N(C(C2CCN(C(CC)=O)C2)=O)CC1 C=CCC(C(=O)N1CCC(NC(=O)CN(CC(C)(C)C)C)C(O)C1)C(C)C C1(CC)CCCC(N=c2nc(N3CCCC(COC)CC3)c3ncccc3[nH]2)C1 C1(CNC(=O)CCN2CCOC2=O)CN(C(c2ncsc2Br)=O)CCO1 N1(CC2CCC(CCC)CC2)CCCC(C)(O)C1 c1(OC(c2nnnn2C)N(CCC)CCN(C)C)ccc(Br)cc1 C=CCC(C(=O)NC1CCN(CCNC(=O)C#CC(C)C)CC1)NC(C)=O N1(C(C(C=C)CC)=O)C(C(=O)N(CC(N)=O)C)CC2CCCC12 N1(C(C(C2CC(NC(CC3(COC)CC3)=O)C2)F)=O)CCC(N=[N+]=[N-])CC1 c1(CN(N2CCC(CN)C2)C)cccc(-c2cnccc2C=O)c1 C1(NC(COCc2cc(CC)no2)=O)CCOCC1C(N1CCC(C)CC1)=O CC#CCC(C(=O)NCC(C)(C)C(C)(F)F)NC(=O)C(F)=CC1CC1 C1(C(=O)NC2CC(F)(CNC(c3c(C)cc(F)cc3)=O)C2)CN2CCCN1CC2 N1(C(CN(C(C(CC)O)=O)C2CCC2)=O)CCCC1C=CC C1(=CC(=O)NC2C(NC(C3(OCC)CCOC3)=O)CCC2)CCCCCC1(F)F c1(C(=O)NC(CC)C(C)O)ccc(CNC(C)=O)cc1 c1(C(=O)NC2CCN(C(CCOCC)=O)C2C)cc(O)nc(C)n1 C1(NC(C2C(C)(CC)C2)=O)C2CCC(C2)C1C(=O)NCCCC(C)(F)F CCC(CN(C)C)C(=O)N(C1CCCC1)CCNC(=O)C(C(C)C)SC N1(C(c2nn(CC)c(C)c2)=O)CCC2CCC(NC(=O)CCc3cn(C)nn3)C12 C1(C)(C(N(CCCCN(C(CCc2c(C)ncs2)=O)C)C)=O)CCCNC1=O C1(=O)CCCCCNC(=O)C(F)CC2CN1C2.C(CN(C)C1CC1)OCC Cc1cc(N(C)CC2CCNC(=O)C2)nc(=NCc2ccc(CO)c(F)c2)[nH]1 C1(C(=O)NC(C)CCNC(=O)CCCn2ccnc2)CC2CCC(C1)N2C1CC1 N1(C(C=COCC)=O)CC(NC(=O)C=Cc2ccc(O)cc2)C(C2CC2)C1 N1(CCCC(=O)NCC2CCC2NC(=O)CC2CCCC2)C(=O)CCC1=O N1(C(CCNC(C)=O)=O)CCC(C)C(NC(C2CC(O)C2)=O)C1 C1(C(N2CCC(CN(C)C)C2)=O)CN(C(c2sccc2CO)=O)CCO1 C=C(C)CC(C(=O)N1CCCCC1CC(=O)N(C)C)OC C1(C)(C(=O)NCC(=O)OCC=C)CCN(C(=O)CCc2cscn2)C1 N1(C(C(CC)C)=O)CCN(C(=O)C(C(C)C)n2cc(C)cn2)C2(CCC2)C1 S(=O)(=O)(c1cccc(C(=O)NC2CCC(=O)NC2=O)c1)Nc1c(C)cccc1 Cc1cccnc1NC(c1nc(-c2cccc(-c3noc(C(N)=O)n3)c2)cs1)=O c1(OC)ccc(N)c(C(=O)NC2CCC2C(=O)NC2(CC(C)(C)C)CC2)c1 Cc1cccc(C)c1CC(=O)NCC1(NC(C2CCOC2)=O)CCCC1 C1(CNC(c2scc(C#N)c2)=O)CC(NC(=O)CC(F)(F)F)C12CCC2 c1(C(=O)NC2C(NC(C(CC#C)C3CC3)=O)CCCCC2)nc2cccnc2s1 N1(C(CCCN(C)C)=O)CCCC(O)(CNC(c2cnn(CCC#N)c2)=O)CC1 CCCC(C)(CC)C(=O)NCC12CC1CN(C(c1nc3ccccc3o1)=O)C2 CCC(C)C(C)(O)CNC(=O)CSCCCOc1ccccn1 C(C(N=[N+]=[N-])C(=O)NC(C)C=CC(=O)NCCOC1CCC1)OCC Cc1ccc(C(CNC(C2CC2C(C)(C)C)=O)NC(=O)Cc2ccccn2)cc1 N1(C(CC(=O)N(C)C)=O)CCC2CC(C1)CN(C(C1CCC(O)CN1)=O)C2 c1(C(=O)N=c2nc(-c3cccc(F)c3)[nH]s2)cc2c(s1)CCNC2 c1(NC(c2cccnc2)CC)ccc(S(=O)(=O)N(CC(C)CO)C)c(Br)c1 C1(NC(c2cc(C)[nH]n2)=O)CC2(C1)CC2C(=O)NC(C)CC(C)C C(=O)(CCCCCC(=O)NC(C)CNC(=O)CCC1CCCC1)OCC c1(CC)ccc(F)cc1C(=O)NC(CNC(C1(CCN(C)C)CC1)=O)CCOC C=C1CCN(C(c2oc(C)cc2C)=O)C(C(=O)NCc2cnc(C)s2)C1 C1(CNC(c2c(COC)scc2)=O)C(C)CCCN1C(c1sccc1C)=O N1(C(c2c(OC)ccs2)=O)CC(N(C(=O)C(C)Cc2cccc(C)c2)C)C(O)C1 C1(NC(CN(C(=O)CN2CCNC(=O)C2)C(C)C)=O)CCC(=O)N(C)C1 c1(C(=O)NCC2CN(C(C3C(C(=O)OCC)C3)=O)C2)n[nH]c2cccnc12 c1(CC)cc(OC)cc(OC)c1C(=O)NCC(C)CN(C)C(C1CCCS1)=O c1(C(N2CC(NC(C3N(C)CCOC3)=O)C(C)(C)C2)=O)cccc2c1nnn2C C=C(C)CC(C(=O)NCCCN(C(=O)CC1CCC(O)C1)CC)NC(C)=O c1(NC(c2n(C=C)nnc2)=O)cc(I)ccc1Br C(C(F)(F)C(=O)NC1CCCN(C(c2ncsc2-c2ccccn2)=O)C1)N(C)C c1(NC(CC(N)C2CCOC2)=O)ccc2c(Cl)nccc2c1 Cc1cccc(C(N2CCC2CNC(=O)Cc2cscc2Br)=O)c1C n1(CCC)ccc(C(=O)NCc2cc(C(=O)NC(C)(CC)CO)n[nH]2)n1 C(C(CC(C)C)NC(=O)CC1CC(=O)NC1=O)NC(Cc1cc(C)sc1)=O C(C1CCOCC1)=CC(N1CCC1CNC1OCCOC1c1ccccc1)=O c1(CC(=O)NC2C(CNC(CNS(CC)(=O)=O)=O)CCCC2)ccc2c(c1)CC2 c1(NCC2(S(C)(=O)=O)CC2)nc(N2CCOC3(CC3)C2)nc2sccc12 Cc1cnn(C)c1C(=O)NC1C=CCN(C(=O)CCc2ccco2)C1 C12(CNC(=O)Cc3cccc(Cl)c3)CCC(CC1)CN2C(c1cnc[nH]c1=N)=O C1(CNC(C(C)(Cl)Cl)=O)CC2CCC(C1)N2C(C12CCC(C)(C1)OC2)=O N1(C(c2c(C)nn[nH]2)=O)CC(CNC(C2CCCC3(CC3)C2)=O)C2(CC2)C1 CCC(F)(C(=O)OC)C(=O)NC1COC2(C1)CN(C(c1ccc(O)nn1)=O)C2 c1(C(N2C3CCC(C3)C2CNC(=O)C(F)(F)C(F)F)=O)cccc2c1CCCN2 c1(OC)cc(C(=O)NCc2ncc[nH]2)c(NCc2ccc(CC(C)C)cc2)cn1 C(=O)(NNc1c(F)cccc1Br)NC1CCCN(S(CCC)(=O)=O)C1 c1(C(N2CCCC(C)(NC(C(C3CCC3)OCC)=O)C2)=O)ccc(S(C)(=O)=O)[nH]1 C#CCCC(N)C(=O)N1CCCCC(OC)C1 N1(S(CCC)(=O)=O)CCC(C(N2CCOC(CC3CCCN3C)C2)=O)CC1 C1(C(N(CC(CN(C)C(c2coc(-c3cccnc3)n2)=O)O)C)=O)CC=CCC1 C1(CNC(C2(CC=C)CCCC2)=O)C2CN(C(=O)CN3CCC(C)C3)CC12 N1(C(C2(C=C)CCN(C(C(C(CC)C)N(C)C)=O)C2)=O)Cc2ccc(C)cc2C1 C1(NC(=O)NC(C2CCSC2)C)CN(C(=O)C(=O)N(C)C)C1 CC(C(=O)NCCCN(C(=O)CSc1nncs1)CCO)=C1CCC1 c1(OC)ccc(C)nc1C(N1CC(CNC(C2(O)CCOC2)=O)C2(CC2)C1)=O n1(C(C)(C)C)nccc1C(=O)NC1CC1NC(C1(Cc2ccccc2)COC1)=O CC(C)C(C(=O)NCCC1CCCN(C(C2CS(=O)(=O)CCO2)=O)C1)C(C)C CCC(CC)C(C(=O)N(CC(N1CCCC1CC(C)C)=O)CC)OC c1(C(N2C(C3CCCN(C(c4cncs4)=O)C3)CCC2)=O)cc2n(n1)CCCC2 Cc1ccc(C(=O)O)cc1S(=O)(=O)NC(=O)CC12CC(C1)C2 N1(C(c2cccc(C(C)=O)c2)=O)CC2CC(C1)CN(C(c1cc(=N)[nH]n1C)=O)C2 C(CCCCCNC(c1ccc(OCC(F)F)nc1)=O)N(C(CC(C)C)=O)C C1(C(=O)OC)CCC2(CCN(C(=O)C(C)(O)COc3ccccc3)CC2)C1 c1(C(N(CCCNC(C(C)NS(CC)(=O)=O)=O)C(C)C)=O)ncc(C)cn1 C1(NC(CCOCCOC)=O)(CO)CCCN(C(=O)Cc2cn[nH]c2)C1 C1(NC(=O)CC2CCOCC2)C2CCC1N(C1C(CS(N)(=O)=O)C1)C2 C#Cc1ccc(C(N2CC(CNC(=O)C(C)C(=C)C)(COC)C2)=O)c(F)c1 C1(C(N2CC(C(=O)NC(C=C)C3CCC3)C(CCC)C2)=O)CC2(CCC2O)C1 C1(C(N2CCC(CCNC(CC3CC(OC)C3)=O)C2)=O)NC(=O)CC1C C1(NC(CCSCC)=O)CN(C(=O)Cn2cnc(Br)n2)C2(CCOC2)C1 c1(COC(c2cc(N)c(F)cc2Cl)=O)ccc(Cl)c2cccnc12 C1(C(N2CCC(O)(CNC(C(COC)COC)=O)C2)=O)CCc2ncccc2C1 n1(C(CC)C)nc(C(N2CCCCC2CN(C)C(C2(C)CC(C)C2)=O)=O)cc1C N1(C(COCC#C)=O)CCC(F)(F)C(CNC(=O)C(O)Cc2[nH]cnc2C)C1 C1(CC)CN(C(c2coc(Cl)n2)=O)CCC1NC(=O)Cc1ccc(C)o1 c1(C(=O)NC2COCCN(C(C3=CCCC3C)=O)C2)ccc2nc[nH]c2c1F N1(C(C(CC)OC)=O)CCC(C2N(C(c3ccc(F)cc3)=O)CC2(C)C)CC1 CC1CCn2c(C(N3CCC(CO)(NC(=O)CCCCC#N)C3)=O)cnc2C1 N1(C(=O)Cn2ccnn2)CCC2(C1)CN(C(C1C3CCC(=O)C13)=O)C2 N1(C(C(C)CC2CC2)=O)CC2COCC(C1)C2NC(=O)C=C(Cl)Cl N1(C(c2cnn(CC)n2)=O)CCCCC1C(C)NC(c1cnc(C(C)(C)C)o1)=O N1(C(c2cc(OC)n[nH]2)=O)CCC(C(=O)NCCC2CC(F)(F)C2)CC1(C)C C1(C(=O)NCC2N(C(C3CN(CC)C(=O)C3)=O)CCC2)CC2(C1)CC(C)(C)C2 C12(S3(c4ccccc4)CN=C4C=CC3=NN4)CC3CC(CC(C3)C1)C2.C1CC1 c1(Cn2c(C(c3cc(C)ns3)NC(CC)CCOC)nnn2)cccc([N+](=O)[O-])c1 c1(-c2cc(C(=O)NC(CNC(C(C)OCC=C)=O)CO)no2)ccc(O)cc1 CC1COC2(C1)CN(C(C1CCN(C(c3ccc(C#N)cn3)=O)CC1(C)C)=O)C2 C1(C(N2CCC(OCCNC(c3nc(C)n(C)c3)=O)C2)=O)CCC2(CCC2)C1 N1(C(COCCC#C)=O)CC2CC(NC(c3cc(Cl)c(C)cn3)=O)CC1C2 C(C(CNC(c1ccnn1C1CC1)=O)C(F)(F)F)NC(COCC)=O C#CC(C)(C)C(=O)NCCN(C(=O)CC(C)CN(C)C)CCCN(C)C c1(N(C2CC3CNC2C3)C(c2cc(C)ncn2)=O)ccc2nc(C)cc(O)c2c1 C1(NC(=O)OC(C)(C)C)CC(O)CN1C(=O)CNc1ccncn1 C1(C(=O)OC)CCOCC1NC(=O)C(c1cn(C)nc1C(F)(F)F)=O c1(NC(CCN(C(C)=O)C)=O)ccnc(Cl)c1I.N12CCOC(C1)CC2=O N12CCN(CC1)C(=O)C1(CCN(C)C1)CC(=O)NCCC2.Cc1sccc1CO C1(CNC(C(C)(C)C2CCCCO2)=O)CCCC2(CN(C(=O)Cc3cnoc3)C2)O1 c1(CC(N2C(CC#N)CN(Cc3ccccn3)CC2)=O)cn2ccccc2n1 C1(C(=O)NCC2C(NC(CSCCCCCC)=O)C2)CCC=CCCC1 CCCN=C(NCC1CCC2(CCC2)C1O)N1CCC(O)CC1 c1(N2CCC(C)SCC2)ncnc2c1ncn2CC(N1CCCCCC1)=O c1(CC(N2CCCCC(NC(C=CC(C)C)=O)C2)=O)nc(F)c(F)cc1F N12CC(F)CC1C2=O.c1(COC(C)=O)ocnc1-c1cn(Cc2ccno2)nn1 CN1CCCCC(C(N2CC3CC3(NC(=O)C=CC3CCCC3)C2)=O)C1=O C12CC(C)CN(C1)C(=O)C=CCOc1ccncc1N2.C(c1ccco1)=CC C1(NC(CSCC(=O)OC)=O)CC2CCC1N(C(=O)C(C)C1CC1)C2 C1(C(N2CSCC2C(=O)NCc2coc(C)c2)=O)(CC)CCNC1=O C(=O)(C1Cc2ccc(Cl)cc21)NC1C(NC(C2CCC(=O)O2)=O)CCCC1 C1(F)(C(N(C(C)CN(C)C(c2sccc2C#N)=O)C)=O)CCCN(C)C1 C1(c2nc(CS(N3C(C(CC)O)CCCC3)(=O)=O)on2)C2CCC1C(OC)C2 c1(OC)ccc(Cl)c(F)c1C(=O)NCCCN(C(=O)CSCc1cscn1)C N1(C(CC(C(C)C)(F)F)=O)CCC2(CCCN2C(=O)CS(C)(=O)=O)CC1 C(=O)(C1CCCc2ncnn21)NC(C)(C)CCNC(C1CC2C=CC1C2)=O N1(C(CSCCC)=O)CCCCC1C1CCN(C(c2snnc2C)=O)C1 c1(C(=O)NCC2CCC(NC(C3CCC(C)CC3)=O)C2)cc2[nH]ccc2s1 Cc1ccc(C)c(C(N2CCC(CN(C)C(C3(C)CC(C)(C)C3)=O)C2)=O)c1O CC(C)C(O)C(=O)N1CCC(C)(CNC(=O)CN2CCCC2)C1 C1(N(C(c2cn(CC)nn2)=O)C)CN(C(c2ccncc2C)=O)CC12CC2 C1(NC(CCCCCOC)=O)CN(C(c2ccc3ccsc3c2)=O)CC1C1CC1 C1(C(C)C)CCN(C(=O)CN(C)C)C(CNC(=O)C(C)C)C1.c12cnc(nc1)[nH]2 C(C(C)C(C)C(=O)NCC1CC(F)(F)CN1C(c1cc(O)nn1C)=O)OC N1(C(C2C(CNC(C=CC=CC)=O)CCO2)=O)CCN(C)C(C)(C)C1 c1(CC)cccnc1C(=O)NC1CCC(C)(CNC(=O)CCc2ccoc2)C1 C(CC[Si](C)(C)C)n1c(C2(NC(C(=O)OC)CSC)CCCC2)nnn1 N1(C(CN(C)C)=O)CCC(C2CCCCN2C(=O)CCC2CC2)CC1 C(CCOC)(C(=O)NCC1CNC(=O)C1)NC(c1cc(CC)sn1)=O Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(c2cnc(N)cn2)=O)CC1O c1(OCC)cc(C(=O)NC2CC2C(=O)NC(C2CCCC2)C)ccn1 CN1CC2(CC(NC(C3CC(NC(c4cc5n(n4)CCC5)=O)C3)=O)C2)C1 CC1=C(C(=O)NCC2CC(NC(=O)C=CC(=O)N(C)C)C2(C)C)COCC1 c1(C(N2C(CCCC)CCC2)=O)cc(C)n(-c2ccc(C(F)(F)F)s2)c1C c1(C(=O)NC2(CCNC(c3c(CC)cc(F)cc3)=O)CC2)cc2c(ccn2C)[nH]1 Cc1nn(C)c(F)c1C(=O)NC1CCC1CNC(=O)C(F)CC1CCC1 Cc1cc(Cl)c(C(N2CCC(NC(=O)CCN3C(=O)CCC3=O)C2C)=O)cn1 C(CNC1CCC(Cc2ccccc2)C1)(CC1CC1)(OC)OC CCCC(C(O)C(=O)NCC1CC=CC1)NC(C1CCC2CC1CO2)=O C1(C(=O)NCc2cc(C)c(O)cc2)CCCN1NC(=O)C(C)C1CCOCC1 N1(C(COCC)=O)CC(C)CN(C(c2ccc([N+](=O)[O-])cc2F)=O)C(C)C1 N#Cc1c(F)c(C(=O)NC2(C(F)(F)C(F)(F)F)CCCO2)cc(F)c1F Cc1cc(CCC(=O)NCC2CC(NC(=O)C(F)C3CCOC3)C2)c(C)s1 C(=O)(CC(C)(C)N(C)C(c1[nH]nnc1C1CC1)=O)NCc1cn(C(C)C)nn1 C1(CC(=O)NCCN(C(CC)C)C)CCCN1C(C1CCC(N(C)C)C1)=O c1(C(N2CCN(C(C3CCCC4(CCC4)C3)=O)CC2)=O)ccc2ncsc2c1 C1(NC(c2csc(C)c2C)=O)COC2(C1)CN(C(C13CC1Cc1c[nH]nc13)=O)C2 Cc1ncnc(C)c1C(=O)NC1CCC(CC(=O)NCC(F)Cl)C1 c1(C(N(CCNC(C2OCCN(C(C)=O)C2)=O)C2CC2)=O)cc(O)nc(O)n1 C#CC1(NS(=O)(=O)CC2CCC(C)N(C(=O)OC(C)(C)C)C2)CCCCC1 C(CCC(C)(C)C(=O)N1CCC(n2ccnc2)C1)NC(CCCCOC)=O C1(C(C(=O)NCC(F)F)N(C)Cc2cc(F)ccc2Cl)CC2(CCCO2)C1 c1(C(N2CC(NC(c3ccc(O)nc3)=O)CC(OC)C2)=O)csc(S(C)(=O)=O)c1 N1(C(C=Cc2c(C)noc2C)=O)CCC2(C1)CN(C(c1ccns1)=O)CCO2 CCC(CC(=O)NCCN(C(=O)CN(C)C)C)CC(F)(F)F C1(CNC(c2cccc(C)c2)=O)CCCN(C(=O)CC2(O)CCC2)CC1 C1(c2nc(C)[nH]n2)CCCCN1C(=O)CC(C)n1cc(Br)cn1 Cc1cc(N2CC(CO)C(C3CC3)C2)n2nc(CO)nc2n1 C12(C(=O)NCCCCCNC(=O)CCF)CCCC1(Br)C2 C1(C(N(CC(C)C)C(C)(C)C)=O)CCCN(C(C2OCCC2(C)C)=O)CC1 C1(CC)CN(C(c2nocc2C(C)(C)C)=O)CCC1NC(=O)C=C(C)C c1(N2CCCC(C(C)NC(=O)Cn3cc([N+](=O)[O-])cn3)C2)cc2nncn2cn1 N1(C(c2c(OC)cccn2)=O)CCN(C(C23CSCC2C3)=O)C(C2CC2)C1 c1(OC)c(NC(=O)NCc2ccc(Br)c(F)c2C)cc(F)cc1Br N1(C(C=C(CC)CC)=O)CCCC2(CCCN2C(C2CCCC3(CC3)C2)=O)C1 c1(C(N2CCC(CC)CC2CNC(=O)CCC2CC2)=O)cc2c([nH]1)CCC(C)C2 c1(CC)oc(C)cc1C(=O)N(CCC(C)NC(C1CCC(C(N)=O)C1)=O)C CCC(C(=O)NC1CCCCCC1C(N1CCOC(C(C)(C)C)C1)=O)C(C)C c1(C(=O)NC2CCC(CNC(c3cc(C)no3)=O)C2)ccc([N+](=O)[O-])cc1C c1(C(C)NC(C2CCN2C(=O)CCC(C)O)=O)nc2ccccc2o1 C12(C(=O)NCCC3(C(N4C(C)CC4CO)=O)CCCC3)CCC(CC1)CO2 c1(NC(=O)CNC(C)=O)ccc(C(=O)COc2ccccn2)cc1 CCC(C)C(=O)NCC(n1cc(C2CC(F)(F)C2)nn1)C N1(C(Cn2cc(C(c3ccc(C)cc3)=O)c(=N)[nH]2)=O)CCC(C)(C)C1C C(=O)(CCCC(C)CC)NC1(CNC(c2c(CC)nn[nH]2)=O)CCCCC1C N1(C(CN=S(C)(C)=O)=O)CCC2(CCCN2C(C2CC(O)C2)=O)CC1 c1(C(N2CCC(N(C(C=CC=CCC)=O)CCO)C2)=O)ccc(F)c(COC)c1 Cn1cc(C2CC2CSC2N(C(N3CCC(CCC(C)(C)C)C3)=O)CCC2)nn1 c1(C(N(C2CCN(C(C3C(CC)C3)=O)C2)C)=O)cncc(N2CCOCC2)c1 c1(NC2CC(NC(C(C(C)C)C)=O)C2)ncnc2cc(C3CC3)nn12 c1(C(=O)NCC(C)N(C(=O)CCC2CC2)CC)cc(C(C)C)n(C)c1C N1(c2nnc(C(=O)OC)o2)CCC2(CCC2)C(NC(c2cncc(OC)n2)=O)C1 c1(C(=O)NC(C(=O)OCC)C)cnc(CCn2cncn2)s1 c1(COC)cc(=NCC(C)(C(C)C)NC(c2sccc2Cl)=O)[nH]cn1 Cc1cc(C(N2CCC3(CC3C(=O)NC3CC(N4CCC4)C3)C2)=O)c(C)cn1 C(CCC(=O)NC(Cn1cccn1)C(=O)NCC=C(C)C)=CC.C1(C)CS1 CC1(C)CN(c2ccc(NC(C3(Br)CC3(F)F)=O)cc2)CCS1 O=C1CC(C2CC2)(C(=O)NCC2CC(CNC(C3CCSC3)=O)C2)C1 C1(NC(CCC(=C)Cl)=O)C2CCC1N(C(=O)C(C)(F)C(=O)OCC)C2 C(=O)(C(C)CC(F)F)N(CC(C)NC(CCCOC)=O)C C12(CCCCC1)C(=O)N2.C1(CC)CN(C(=O)CC2CCC(C)C2)CCO1 C1(NC(C2(CN(C)C)CC2)=O)CC2CC(NC(=O)CCc3cc(Cl)cs3)CC2C1 c1(C(N2C3CCC2CN(C)C3)C(=O)NCC)ccc(Cl)c(Cl)c1Cl c1(C(=O)NCCCCCC(=O)N(C2CC(C(=O)OC)C2)C)cc[nH]c2nccc1-2 N1(C(Cc2nc(C)sc2C)=O)CCCC(C)C1CNC(=O)CCCC1CCC1 C1(C(=O)NCC(CN(C)C(C2CC2c2cccnc2)=O)O)CCCC1C(N)=O c1(C(=O)NCC2(CCNC(C(C)NS(C)(=O)=O)=O)CC2)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2CCCC(NC(C(C#C)(C)C)=O)CC2)cc([N+](=O)[O-])c(C)cc1C N1(C(C(C)NC(C)=O)=O)CC2C3CCC(C2C1)N(C(c1cnc(CN)cn1)=O)C3 c1(OC)c(Br)ccc2ncccc12.c12cc(Br)ccc1c1c[nH]nc1c(=O)[nH]2 c1(C(=O)NC(C(=O)NC(C)C(C)C)Cn2cccn2)cc(O)ncc1F C1(C(NOCC(=O)NCCN(C(C)C)C(C)C)=O)CC2CCCC2C1 c1(C(N2CC(C)(C(=O)Nc3c(O)ccc(CC)c3)C2)=O)cccc2c1CCCC2 c1(C(=O)NCCCCN(C)C(C2CCCC(=O)N2)=O)cccc2c1CCO2 O=C(Cc1ccccc1S(=O)(=O)N1CCCNCC1)N=c1ccc(Cl)n[nH]1 CC(C)CC(C)(O)C(=O)N1CCC2(CC1)CC2NC(=O)CC1CC1 CC1(C)CCC(Cl)=C(C(=O)NC(c2ccccc2)c2cccnc2)C1 c1(N(C)C)noc(C2c3ccc(C(N)=O)cc3C(=O)N2C2CCC([SH](=O)=O)C2)n1 Cc1cc(CC(=O)N(CCCN(C)CC2CCCS2(=O)=O)C)cc(Br)c1 CCCCC(F)C(=O)NC1CCOC(C(N2CCC2CC)=O)C1 N1(C(Cc2c(C(=O)OC)cccc2)=O)CCN(C(C2CC2C)=O)CC1C C1(c2ccn(C3CN(C(C4CCCO4)=O)C3)n2)(NC(=O)NC(C)C)CCCC1C c1(NC(C=C)C)nc(N2CC(C#N)C3(CCC3)C2)nc2c1ncn2C N1(C(c2ncn(CC)c2)=O)CCCC(N(C)C(c2cc(C3CCC3)nn2C)=O)C1 C1(C(=O)NC(C)CCCCNC(c2cnn(CCF)c2)=O)CCc2n[nH]cc2C1 Cc1cccc2[nH]cc(CNc3ccc(C(C)C)cc3)c12 n1(CC=C)nnnc1C(c1cnn(CCF)c1)NCCCCF N1(C(c2c(N)cncc2)=O)CC2(CCC2NC(=O)Cc2cnns2)C1 c1(OC)cc(OC)cc(NC(=O)C(C)NCC(c2ccccc2Br)O)c1 Cc1ccc(CC(=O)N(CC(C)(C)NC(=O)C(F)C2CCC2)C)cn1 N1(C(CC=C)=O)CCc2c(C(=O)NCC(C)N(C)C)cccc2C1 C(=O)(CCCCC(C)(C)C)NC(CN(C(=O)C(O)C(F)(F)F)CC)C CCCC(C)CCCC(=O)NC1COCCN(C(=O)C=CC(=O)OCCCC)C1 C1(C(N2CCCC(C(C)C)C2)=O)C(C2CC2)CCN1C(c1csc(O)n1)=O C1(C(N(CCOCCOC)C)=O)CN(C(=O)C(C)n2cnnn2)CC(C)O1 CC1(C)C2CCC(CN3C(=O)CN(CC4CCCCCC4(F)F)C3=O)C1C2 C1(C(N2CC(CN(C)C(C3CS(=O)C3)=O)C3(C2)CC3)=O)CCOCC12CCC2 O=C(C(O)Cc1ccccc1Br)N(C1(c2cn(CC(F)(F)CO)nn2)CCC1)CC N1(C(C2(C)CCOCC2)=O)CCCC(NC(=O)COCC2CCCC2)C(F)C1 N1(C(C(C)OCCOCC)=O)CCC(C2(NC(c3ncc(Cl)s3)=O)CC2)CC1 c1(C(=O)NCC2N(C(C3C4(CC(C)OCC4)C3)=O)CC2)cc2cc(N)ccc2o1 N1(C(C(COC)O)=O)C2CCCC1CN(C(c1cccn3cc(C)nc13)=O)C2 c1(NC(C)=O)cccc(C(=O)NCC(C)N(C(=O)Cc2ccns2)C)c1C c1(C(N(C(C)CNC(=O)C(n2ccnc2C)C)CC)=O)cnc(O)cc1C C(=O)(CC(O)C(Cl)(Cl)Cl)NC1(CC)CCCN(C(=O)CN(C)C(C)=O)C1 N1(C(C2(CO)CCC2)=O)CCC(Cn2cc(CC(O)CO)nn2)C(F)(F)C1 C1(C(=O)NC(C2CC(NC(C(C)C)=O)C2)C)CC2(CCC2O)C1 Cc1cc(C(N2CC3CN(C(C4CCC(C(C)C)CC4)=O)CC23)=O)cc(C#N)c1 CC(C)(C)C(C)(C)C(=O)NCC(CO)NC(=O)COc1ccc(F)nc1 c1(NC(CN2CCN(C(C(C(C)C)=O)=O)CC2)=O)cc2ncnc(O)c2cc1Cl c1(C(N2C(C)(C)C(C(=O)NCC3(CC(N)=O)CC3)CC2)=O)cc2ccncc2[nH]1 Cc1cc(=NCc2cc(Br)cn2C)[nH]c(NC2CCC(O)CC2)n1 c1(-c2scc(C(=O)NC3C(CNC(C=C(COC)C)=O)C3)n2)ccc(F)cc1 c1(C(=O)NCCC(C)NC(c2cnn3c2OCC3)=O)cc2n(c1)CCCC2 CCC(C)C(CC(=O)Nc1cccc(O)c1)NC(=O)C(O)CCC(C)C N1(C(CC(=O)OC)=O)CCC2CCN(C(=O)Cc3ccc4ocnc4c3)CC2C1 c1(NC(c2c(NC(c3ccn(C)n3)=O)cccc2)=O)cc2n(n1)CCC2 C(CC(C)(C)C)(C(=O)N(C1CC(NC(c2cnc(Cl)c(N)c2)=O)C1)C)OC C12CCCN(CC1)C(CC)C(=O)N2.C=CCCCC(=O)NC1C(N(C)C)COCC1 N1(C(c2c(C(=O)OC)ccs2)=O)CCC(F)(C(=O)NCC(O)CN(C)C)C1 N1(C(c2c(C)nncc2)=O)CCC2CCN(c3cc(O)nc(O)n3)CC2C1 c1(OC)ccc(O)c(CN2C3CC2CN(C(=O)CCc2cnn(C)c2C)C3)c1 N1(C(C2CC(F)CCN2C(=O)CSC2CC2)=O)CCCC(c2ccncc2)CC1 C(CO)(CCCCNC(C1(C)CCN(C)C1)=O)NC(C1(CC=C)CC=CC1)=O Cc1nc(O)nc(C)c1CC(N1CCC(=CCNC(C2C(C)C2(F)F)=O)CC1)=O C1(O)(CN(C)C(c2ccccc2C2CCC2)=O)CCN(C(=O)Cc2ccon2)C1 CN1Cc2ccccc2CC1C(N1CSCC1c1nn[nH]n1)=O C1(NC(c2n(C)ccc2)=O)CC2CN(C(C3CCC(C)(F)CC3)=O)CC12 c1(-c2cc(C(=O)NC3(CNC(CCOCC)=O)CCOC3)on2)ccccc1Cl C(=O)(CCC(=O)NN(C)C)N(CCOC)CCNC(=O)Cc1ccccc1C C1(CNC(C(C)NC(c2cccs2)=O)=O)CCN(C(c2ccnc(F)c2)=O)CC1 n1(CC)cc(C2OCCC2CN2CCC2c2nccn2C)cn1 c1(NCC2(C)CCCOC2)nc(=NCC2(S(N)(=O)=O)CC2)[nH]c2cc[nH]c12 C(=O)(CCC(C)(C)N(C)C)N1C(C(C)NC(=O)CC(O)CN(C)C)CCC1 C1(C(=O)NCC(C23CCC(CC2)C3)NC(C=CCOC)=O)CCN(C)C1=O c1(C(C(=O)NC(C)CCC2CC2)NC(COCCOCC)=O)ccc(Cl)cc1Cl c1(C(=O)NC2CC(CNC(C3C(CC(C)C)C3)=O)C2)ccc2c(c1)NC(=O)C(C)O2 N1(C(CC(=O)NCC2CC2)=O)CCCC(CO)(NC(c2cc3sccc3[nH]2)=O)C1 c1(C(=O)NCC(C2(O)CCN(C(c3ccc(O)nc3)=O)C2)C)cc(Cl)ccn1 C1(CC)C(C(=O)NCC2C(C)(C)C2(F)F)CCN1C(c1cn(C2CC2)cn1)=O C(=O)(C1=NOC2(CCC2)C1)NCC1C(C)CCN(C(c2cc(C)n(C)n2)=O)C1 N1(C(c2c(SCC)ocn2)=O)CCC(C(=O)NCC2CCC(=C)C2)CC1(C)C C(=O)(CC(C)CCC(=O)N1CCC(CNC(C2C=CC=CC=C2)=O)C12CC2)OC CC1(C)CN(C(=O)CCc2ccccc2O)CCN(C(=O)CC2C=CCC2)C1 c1(NC)snc(C)c1C(=O)NCC(C)(C)CNC(c1ccc(OCCO)cc1)=O CN1CCCC(c2cccc(C(=O)NCC(F)CNC(C3(C#N)CCC3)=O)c2)C1 c1(SCC(NNC(c2nn(C)c3c2cccc3)=O)=O)ccc2c(c1Cl)OCCCC2 c1(C(=O)NCC2(C)CCN(C(c3cnc(F)c(F)c3)=O)C2)ccnc(Cl)c1Cl Cc1cn(C(C)C(=O)N(C)CCOCCNC(=O)Cc2nc(C3CC3)no2)nn1 c1(OC)c(C)cc(C(=O)NCC2CN(C(=O)CCCCC3CC3)C3CC23)cc1C CC1(C)CC1(C)NC(C1CCCN1C(=O)CC1COCCO1)=O c1(C(=O)NC2CC(C)(NC(=O)CCC(C)(F)F)C2)ccc2c(c1)OC(C)(C)O2 N1(C(C(C)c2cccs2)=O)CC(C)(CCC(=O)N(C)C)C1.C1CC(=O)N1 O=C(CS(=O)(=O)Cc1cccs1)NC1CCC(NC(=O)CCCN2CCCC2)C1 Cc1cc(C)n(C(C)CNC(=O)Nc2cc(CSc3ccccc3)ccn2)n1 c1(OC)cnc(C(N2CC3C(CNC(=O)CSCCC(N)=O)C3C2)=O)nc1 CCCCC(C(=O)N1CCSC(C(C)C)C1)NC(c1cn(C2CC2)nn1)=O C1(CC(=O)NCC(CNC(c2cc(C(C)C)no2)=O)O)CCCC12CC2 N1(C(C2C3(CN(C(COCC(=O)OC)=O)C3)C2)=O)CCC2(CNC(=O)O2)C1 Cc1cc(N2CC3CCC3(C)C2)nc(N(C2CCOCC2)C)n1 C1(O)(c2cn(C(C)C3CC3)nn2)CCCN(C(C2CCCC(O)C2)=O)CC1 c1(C(N2CCC(NCc3c(Br)ccc(C)c3)C2)=O)c(O)cccc1[N+](=O)[O-] CC1(C)CCN(C(=O)COC(F)(F)F)CC1NC(C1CCOCC1(C)C)=O Cc1cc(C(N2CCC(NC(C3CCN(C)C3)=O)C(F)C2)=O)cnc1C c1(C(=O)NC(c2ccnn2C)C(=O)NCCc2onc(C)n2)ncc(F)cc1N Cc1coc(C(=O)NCCC2(NC(c3cc(F)n(C)n3)=O)CC2)c1C c1(C(=O)NC(CC)CN(C(=O)CSC2CC2)C)ccc(C)n(C)c1=O O=C(C1CCc2cccc(=O)n21)NC1CN(C(=O)CCc2cc(Cl)cc(Cl)c2)C1 Cc1nc(C(=O)NC(CO)C(C)C)sc1-c1ccc(-c2ccc(F)cc2)cn1 C1(C(=O)NCC2CC(CNC(Cc3cc(C)no3)=O)OC2)CC=CCC1C C12(NC(=O)NCCCCC)CCN(C(c3ccc(OC)cc3)=O)CC1C2 Cc1cc(C(=O)NCCCCc2ccc(Cl)cc2)n(C(C)(C)C)n1 C1(CNC(c2c(C)cc(CO)o2)=O)C(C)CCCN1C(=O)Cn1cccn1 c1(N2CCC(CC)C2)ccc(S(=O)(=O)NCC2CCCN2C)cc1C#N N1(C(c2c(C)cnn2C)=O)CC2CC(NC(=O)CCc3cccnc3Cl)CC1C2 CC1CCN(C(c2ccnc(F)c2)=O)CC1NC(=O)CO Cc1c(C(N2C3CN(Cc4ccc(Br)c(C(F)(F)F)c4)CC23)=O)cccc1O CS(=O)(=O)C1(C(N2CC(NC(=O)C=Cc3cscn3)C2)=O)COC(=O)C1 N1(C(C(F)OC)=O)CCC2(CCCN2C(c2cc(Br)cnc2O)=O)C1 Cc1[nH]nc(Cl)c1C(=O)NCCC(C(C)C)NC(C1CC2C=CC1C2)=O c1(C(c2nnnn2C(C)(C)C)NC(C(=O)NCC)C)c(C)cc(Br)cc1F C1(C(N(c2cn(C(C)C)nc2)C)=O)COCCN(C(C2CCCCCCC2)=O)C1 C(=O)(C(F)CCC(C)C)N(C(CNC(c1c(C)c(C2CC2)[nH]n1)=O)C)C N1(C(c2ccccn2)=O)CCCCC1Cn1cc(CCC2CCOC2)nn1 c1(CCCN2CCN(c3cc(F)cc(Cl)c3)CC2)nc2ccccc2[nH]1 C#CCC(C)C(=O)NCCc1ocnc1CNC(C1CC1c1cccc(F)c1)=O N1(C(C(c2cccc(F)c2)C)=O)CC2(C)CN(CC3CCC(C)CC3)CC2(C)C1 c1(N2CC(CNC(C(=C(C)C3CC3)F)=O)C(C)(C)CC2)ncc(C)cc1[N+](=O)[O-] Cc1ccc(C(=O)NC2(C3CN(C(=O)CCCc4cnccn4)C3)CC2)cc1O N1(C(C(CC(=O)OC)C)=O)CC2CN(C(c3cc(F)c(Cl)cc3Cl)=O)CC2(C)C1 c1(C(=O)NC2CC(C)(CNC(C3CCC(F)C3)=O)C2)cnn2c1NCCC2 C1(C2CCCCC2)CCN(N2CCC2c2nc[nH]n2)C2(CC2)C1 C12(C(N(c3cccc(NCc4ccccn4)c3)C)=O)CCC(C(F)F)(C1)OC2 C12(NC(Cc3n(C)c(S)nn3)=O)COCCC1CN(C(c1ncccc1Cl)=O)C2 C1(C(Cn2cc(-c3n(C(C)C)ccn3)nn2)F)CCN(C(=O)C(C)(Cl)Cl)CC1 CCCCC#CC(C)(C)NC(=O)C(c1ccco1)NC(C1CC(=O)N(CC)C1)=O C(c1ccncn1)=CC(=O)NC(c1cn(C)nc1)C(=O)NCC1CC(O)C1 n1(CC(=O)NC(CNC(C(C)OCC#C)=O)(C)CO)nc(C(F)F)cc1C1CC1 N1(C(C(C)CO)=O)CCC2(CCOCC2)C(NC(c2cccc(S(C)=O)c2)=O)C1 C12(NC(c3cc(OC)ns3)=O)CCC(CC1NC(c1cccc(C)c1O)=O)C2 c1(C(=O)NCCC(C)(C)NC(C=CCC)=O)ccc([N+](=O)[O-])cc1 C#CC(CNC(=O)C(C1CN(C(c2ocnc2CC)=O)C1)OC)C(C)C C12(CNC(C3(C#C)CC3)=O)CCC1CN(C(=O)CCc1c(C)noc1C)C2 CC1(NC(c2ccncc2Cl)=O)CCCCC1C(=O)NCCC1=CCCCC1 CCC(C)(C#N)C(=O)N1CC(O)(CNC(c2ccc(C)c(Br)c2)=O)C1 N1(CCCC(=O)NCCNC(Cn2ccc(C)n2)=O)C(=O)c2ccccc2C1=O N1(C(CCC(C)=O)=O)CC(C)(C)CCC1CNC(C1(C)CC(C2CC2)=NO1)=O c1(C(=O)NCCC2CCN(C(=O)C=CC(F)(F)F)C2)ccc2nc(Cl)nn2c1 CCCCCCCC(=O)NC1CCC12CN(C(=O)C(=Cc1c[nH]cn1)F)C2 N1(C(c2onc(CC)n2)=O)CCCCC(NC(=O)C=Cc2nccn2CC)C1 S(=O)(=O)(c1cc(F)c(Br)c(F)c1)N1CC(C(=O)Nc2cn(COC)nc2)NCC1 C(c1ccnn1C)=CC(=O)NCC=CCC(=O)NC(c1cnn(C)c1)C N1(C(C2(CC(C)C)COC2)=O)CCCC(O)(CNC(C2CC(F)(CO)C2)=O)C1 C(C1OB(O)c2ccccc21)N(C(=O)CC1CCC2(CC(C(=O)O)C2)O1)CCO c1(C(=O)NCC2CC(NC(CC=C)=O)C2)cccc(SC(F)(F)F)c1 c1(C(=O)NC2CN(C(C3(CC=C)COC3)=O)CC2O)cc2c(C)cc(F)cc2[nH]1 CC1COCC(CNC(=O)Cc2nncs2)O1 c1(CC(N2CC(CNC(CC=CCC)=O)(COC)C2)=O)c(F)cc(F)cc1F Cc1ncc(C(N2CCC(C(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)c(C2CC2)n1 c1(C(NOCC#C)=O)ncoc1CNC(C1CC1C(C)(F)F)=O CC(C(=O)N1CCC1CC(=O)NCC12CCCN1CCC2)S(C)(=O)=O CCCC(CCCNC(=O)CC1CCN(CC)C1)NC(=O)CCc1cncn1C N1(CCC(=O)N(CC(C)(C)CNC(c2ccccc2)=O)CC)CCS(=O)(=O)CC1 N1(C(=O)OC)C(C)CN(C(=O)COC(C(C=CC)O)=O)CC1C C=CCC(CC(=O)N1CC(N(C)C2CC2)C1)NC(=O)C(C1(O)CCCC1)F n1(CC(C)NC(=O)CN2CC3CC3C2)cc(CN(C)C)nn1 C1(NC(COCCCOC)=O)CCN(C(=O)CCOCc2nccn2C)C(C)C1 c1(C(NNC(Cc2c(OC)cccc2)=O)=O)nc2c(s1)CCCC2 Cc1nc(N2CCC(F)(CNC(=O)CCS(C)(=O)=O)CC2)cc2nncn12 N1(CC(C)C)CC2CCN(C(c3ccsc3-c3nn[nH]n3)=O)CC2C1 C1(CNC(CC=C(C)C)=O)C2CN(C(=O)CNc3ccccc3C(N)=O)CC12 c1(C(N(CC(=O)NCCCNC(N)=O)CCN(C)C)=O)cccc(O)c1Cl CC(C)(C(=O)NCC1C2CCC(C2)N1C(=O)CNC(c1cccs1)=O)S(C)(=O)=O C(=O)(C(CNc1cc(Cl)ccc1C)C(C)(C)C)N(CCOCC)C N1(C(c2cncc(CC)c2)=O)CCN(C(=O)CCn2ccc(C)n2)CC12CC2 C1(C(=O)NCC2CCN(C(C3(C(C)C)CCC3)=O)C2)CCCCC1n1ccnc1 c1(C(=O)NC2CCCN(CC#N)CC2)cc(Br)cn2ncnc12 C(=O)(CC1=CCN(C)CC1)NC1C(NC(c2ccc(C)o2)=O)CS(=O)(=O)C1 CC1CCCC(C(=O)NC2(C)CCCN(C(C3CC(O)(C(F)F)C3)=O)C2)CC1 c1(NC(C#C)(C)C)cc2sc(C)cc2n1CC(=O)OC(C)(C)C c1(C(N2CC(CNC(C(CC)C#N)=O)C3(C2)CCC3)=O)ccc2c(c1)CCCC2 C1(C(=O)NCc2ncc[nH]2)(NC(C2(Cl)C(C(C)=O)C2)=O)CC(O)C1 C=CCCN=C(NCC1CC(N2CCCCC2)CCO1)N1CCCC(N(C)C)C1 Cc1scc(C(=O)NCC(C)N(C)C(C2CC2C(N)=O)=O)c1N C1(NC(c2ccnc(Br)c2)=O)CC(NCc2nc(Cl)sc2Cl)C12CCC2 N1(C(c2c(CCC)[nH]cc2)=O)CCCC(CCNC(c2ccncc2Cl)=O)CC1 C1(=CC(=O)NCC(C2CC(c3nn[nH]n3)C2)=O)CC2NCCC12 C1(NC(CC2(C)CC(F)(F)C2)=O)CN(C(C2CCOC(=O)CC2)=O)C2CCCC12 c1(NC(N2CCC(c3cnc(OC)c(C)c3)CC2)=O)ncc(S(=O)(=O)C(F)F)cn1 C1(O)(CNC(=O)CSCc2ncc[nH]2)CCN(c2nncs2)C1.C1(C2CC2)(N)CC1 O=C(CCC(F)F)NC1CCCN(C(=O)C(Cc2ccccc2)C2CC2)C1 C(=O)(C(F)C(=O)N1CCC(C)(CNC(c2c[nH]nc2CC)=O)C1)OCC c1(C(N(C(C)CNC(=O)CCc2cccs2)C)=O)ccc(C(C)(C)C)o1 C1(NC(c2ccc(OCCC)cc2)=O)CCN(C(C2(CC)CCCO2)=O)CC1O N1(C(C(CC)SC)=O)CCC(CC(=O)N(C)Cc2scnc2C)C1(C)C c1(CC(F)(F)F)cccc(NCc2ccc(Br)cc2)c1 c1(C(=O)OC)cc(C(N2CCOC(CNC(=O)C3=CCCO3)C2)=O)c(C)o1 c1(OCC)ccc(C(=O)NC2CC(C)CN(C(=O)CC3(C)CCCO3)C2)cc1C C1(NC(c2ccc(CC)o2)=O)(CO)CCCN(C(=O)CCc2nc(O)n[nH]2)C1 c1(C(N2CCCC(CCC)(NC(=O)CN(C)C3CC3)C2)=O)ccc2ccoc2c1 N1(C(C(COC)OC)=O)CC(C)N(C(=O)CCn2nc(C)nc2C)CC1C c1(NCC2(C)N=C(C)SC2)cc(N2CCC(N3CC(=O)NC3=O)CC2)nc(C)n1 c1(CC(=O)NCC(CC=C)NC(=O)Cc2cc[nH]n2)ccc2oc(C)nc2c1 Cc1c(C(N2CCC(C(C)C(=O)NCc3cnco3)C2)=O)cncc1F N1(C(c2ccc(N(C)C)nc2)=O)CC2CC3CC2C1C3NC(=O)CP(C)(C)=O Cc1c(C(=O)NC(C)CNC(c2cc(Br)co2)=O)cccc1F C(=O)(C1=CCCN(C(C2CCCOC2)=O)C1)NCc1cnc(C(C)C)[nH]1 c1(C(N2CCC2(C)C(C)C)C(=O)Nc2c(C)cccc2)ccc2c(c1)OCC2(C)C C1(C)(C(N2C3CN(C(CC4CCC(C)CO4)=O)C(C3)C2)=O)CCC(F)(F)CC1 C1(N(C(CC2(CC)CC2)=O)COC)CCC(CNC(=O)C(C2CCCC2)OC)CC1 C(CC(=O)N1CCCC(CO)C1)(C(F)F)NC(c1ccn(C)n1)=O n1(CC(=O)NCC2(C)N(C(C(C=C)(F)F)=O)CCC2)cc(C#N)c(O)nc1=O C1(C(=O)NCC2C(NC(CSCc3ccc(C)cc3)=O)C2)OC2CCC1CC2 N1(C(COCC(C)(C)C)=O)CCC2(CCC2NC(=O)CNS(N)=O)CC1 C1(NC(C2(C)CCOC2)=O)CN(C(C2(c3cccc(N(C)C)c3)CC2)=O)CC1O N1(Cc2n(CCC)ccn2)CCN(C(C2CC23CC3)=O)CC1 N1(C(C(N)=O)=O)CC(NC(=O)CCCF)CC2(CCOCC2)C1 c1(CC)ccc(C(=O)NCC(O)CN(C(=O)C(F)(F)c2ccnn2C)C)c(N)c1 C1(O)(CCNC(c2c(CC)cns2)=O)CCN(C(=O)CN2CCCC2C)CC1 CC1(CNC(C2(C)CC2(Cl)Cl)=O)CCN(C(=O)Cc2csnn2)C1 N1(C(C(C)NC(c2cscc2F)=O)=O)CC2CC1C2NC(C1CCCCC1)=O CCCC(CC)C(=O)N1CC(CNC(c2cn(CC3CC3)nn2)=O)C(O)C1 C#CC1(O)CCN(C(C2CC23CCN(C(c2cnnn2CC)=O)C3)=O)C1 C=C(CNC(C1CCC1)=O)CCNC(=O)CCc1ccc(Br)s1 C1(CC)CN(C(c2ccc(Cl)s2)=O)CCN1C(c1ns[nH]c1=O)=O c1(-c2onc(C)n2)ccc(NC(=O)C(=O)NCCc2ccsc2)cc1 c1(C(=O)NC2CCC3(CN(C(CCCC=C)=O)C3)C2)ccc2c(Br)c[nH]c2c1 C1(NC(COC)=O)CN(C(=O)CC(CN(C)C)C(F)F)CC2(CCC2)C1 n1(CC(=O)NC2C(NC(c3cccc(OC)c3)=O)CC2)cccc([N+](=O)[O-])c1=O C1(C2CCC2)(C(N2C(C)CCC(CNC(C3CCCS3)=O)C2)=O)CC1(F)F N1(CC(=O)NC2CC3(CN(C(c4c(OC)scc4)=O)C3)C2)CCc2ccccc21 CC(c1ccccc1F)=CC(=O)NCC(CO)NC(=O)CC1CCCC(=O)N1 N1(C(CN(CCC)C)=O)CCCC(C)(C)C1CNC(C1(C)CC(F)C1)=O C(C(N=c1ncnc2[nH][nH]c(C)c1-2)C1CC1)NC(C1N(C(CCC)=O)CCC1)=O N#CC1(C(N2CCC2C(=O)NCCc2cc[nH]n2)=O)CC(=O)C1 c1(CC(=O)NOCC2CCCS2)ccccc1Cl c1(CC(N2CCN(C(Cc3nc(C)on3)=O)CC2CO)=O)ccc2ocnc2c1 N1(C(CCC)=O)CCC(N(C(C23CCC2C3)=O)Cc2ccccn2)CC1 C1(C(N2CC(OC)(CNC(=O)Cn3cc(Cl)cn3)C2)=O)CCCN(C(N)=O)C1 Cc1cc(C)cc(C=CC(=O)NCCOCCCNC(C2CCCNC2=O)=O)c1 C(=O)(C(F)C(C)(F)F)N(C1(CCCC(=O)NC(c2cnccn2)C)CC1)C c1(CC=C)ccc(C(=O)NCC2COCC2NC(c2coc(COC)n2)=O)cc1 CC(C)C(CNC(c1cccc[n+]1[O-])=O)C(=O)N1OC2CC1C(O)C2O Cn1cc(N)c(C(N2CCN(C3CN(C(=O)C=CC4CCC4)C3)CC2)=O)n1 C1(NCc2c(Cl)cncc2Cl)CCC2(CC1)CCOC2 c1(N2CC(C(C)NC(=O)CC3CC(O)C3(C)C)OCC2)ncnc2c1CCCC2 C(C(C)(O)CC(=O)N1C(C(=O)NC(CO)CCCO)CC2CC12)OC C(=O)(C1=CCOCC1)N(CCC(C)NC(c1ccc(C(C)=O)nn1)=O)C CC(C)(CNC(c1nnnn1C1CCCCC1)c1ccsc1)CC1CCCC1 N1(C(CC2(CC)CCC2)=O)CCOCC1(C)c1cn(CCOC2CCC2)nn1 c1(C(=O)NCCOC2CN(c3ccnc(C4CC4)n3)C2)cc2c(s1)CCOC2 N1(CC(=O)NC(C(C)NC(C2CC(C(=O)OC)C2)=O)CO)CC2CCC1C2 N1(C(c2ccn(COC)n2)=O)CCCCC(CNC(C2CC3(CSC3)C2)=O)C1 CCC1=C(C(=O)N2CC(C3CN(C(c4cnn(C5CCC5)c4)=O)C3)C2)CCCO1 N1(c2c(OC)nccc2)CCC(O)C(C(=O)NC(c2nc(C)cs2)C)C1 c1(C(N2CC(CNC(=O)CC3CC4(COC4)C3)OCC2)=O)nsc2ccccc12 c1(CC)ccc(F)c(C(=O)NCC(N2CCN(C(C3(C)CCCS3)=O)CC2)C)c1 C1(NC(CC(C)(C)SC)=O)CC2CCC1N(C(C1(NC(C)=O)CCC1)=O)C2 CC(C)(C)C(CNC(c1ccc2c(Br)cnn2c1)=O)CC(=O)O C(CC(C(=O)N1CC(CNC(=O)CCc2nccs2)C(C)C1)NC=O)SC Cc1ccc(C(=O)NC(CNC(C2CCCCCC2)=O)C2CC2)c(C(C)C)n1 C1(OC)CC(NC(c2cnc(O)n2C)=O)CN(C(c2ccnn2CCF)=O)C1 c1(C(=O)NCC(CC(=O)OC)C(F)F)cc([N+](=O)[O-])c(C)cc1C C1(C)(CCNC(C(CC)C)=O)CCN(C(=O)COC(F)(F)F)C1 C#CC1(C(=O)NCCC2CCOC2)CCN(C(c2cccc(O)c2F)=O)C1 CCC1=NOC(C(N2CCC(C(C)NC(c3n[nH]cc3F)=O)CC2)=O)C1 c1(C)cccc(OCCN)c1OC.C(=O)(COCCF)N(CC=C)CCO.N c1(C(N(CCNC(=O)COCc2ccncc2)CC)=O)cc(C)c(F)cc1Cl Cc1cccc2cc(CNC(c3cnn4ccccc34)C)sc12 c1(CC)nc(C(=O)NCC(CC)NC(c2cnoc2-c2cnn(C)c2)=O)co1 C1(C(=O)NCC2CC(CNC(c3cn(CC)nn3)=O)C2)CCCS(=O)(=O)C1 C(c1cccc(Br)c1)=CC(N1CC(CCNC(c2ccc(Cl)cc2)=O)C1)=O C(=O)(C(O)CCSC)N(CC(=O)NCCc1ccc(C)cc1)CC#C C(C(F)(C(=O)NC1CCCN(C(C)C)C1)C(C)C)NC(COCCOC)=O N1(C(C(C)Cc2ccccn2)=O)CCC(C(N2CC(N(C)C)C2)=O)C(C)C1 Cc1ccc(Cl)c(OCC(=O)NC2CC(NC(C3(O)CCCCCC3)=O)C2)c1 N1(C(C(C(C)(C)C)=O)=O)CCN(C(=O)C=Cc2ccco2)CC(O)C1 C1(CN(C)C)CCCN(C(c2cc(CCCOCC(=O)NC3CC3)no2)=O)C1 CC(CCNC(=O)Cn1cnc(C(F)(F)F)n1)CCNC(c1cccnc1N)=O C=C(C)CC(C(=O)N1CC2C=CC1CC2)NC(C1C(O)C2CCOC12)=O C(=O)(CC(C)C(=O)NC(C)CNC(c1cc2n(c1)CCC2)=O)OC N1(C(C=CC(C)NC(=O)CSC(F)F)=O)CCN(CCO)C(C)C1 C1(C)(CCNC(CNC(C(C)(C)C)=O)=O)CCN(C(c2cccc(Cl)c2)=O)C1 Cc1nc2cc(OC(C)C(N3CCCC3C(C)C)=O)cnc2[nH]1 c1(C(=O)OCc2cn(CC)nn2)ccc(-c2nnco2)cc1 c1(C(N(CC(C)NC(CCCc2cc(C)no2)=O)C)=O)ccc(C#N)nc1O c1(CC)occ(C)c1C(N1CCCCC1CN(C(=O)CCCOC)C)=O C1(OC)CN(C(c2ccnn2CCF)=O)CCC1NC(=O)CCC1CCC(=O)N1 c1(C(C)(C)C)cccc(CNC2CC(F)CN(C(c3sccc3F)=O)C2)c1O C1(C2CCN(C)CC2)(C(N2CC3(CN(C(c4c(C)cnn4C(C)C)=O)C3)C2)=O)CC1 c1(CC)onc(C)c1C(N1CC2CC1C2CO)=O.c12c[nH]nc1C(=O)NC2 N1(C(c2cc(Br)cs2)C(=O)NCC(C)C)CCN(CC)CC1.C(C)(C)(C)OC(=O)NC Cc1nn(C)cc1C(C)NC(=O)NCC1CC(F)(F)C1 C(=O)(CCS(C)(=O)=O)NCCn1ncc(C(N2C(C#C)CC2)=O)c1 C1(NC(C(C)SC)=O)CCN(CCC(C)F)C1 c1(C(=O)NCC(CN(C)C(c2nnn3c2CSCC3)=O)O)ccc2nccn2c1 c1(C(=O)NC2CN(C(C=CC(=O)N(C)C)=O)CC2O)cccc(O)c1F c1(C(N2CC(C)=CC(C)C2)C(=O)NCC)ccc(F)c(Br)c1F c1(C(N2CCC(C(C(C)C)NC(C(C)SC(C)C)=O)CC2)=O)cccc(Cl)c1F C1(C(=O)NCC2(OC)CN(C)C2)C(C2CC2)CCN1C(=O)CC1CC(OC)C1 c1(CC(=O)NC2CCCC(NC(C3(O)C(C)(C)C3)=O)C2)nc(F)c(F)cc1F Cn1cnc2c[nH]c(=NCC3(C)CCN(C(c4n[nH]cc4[N+](=O)[O-])=O)C3)nc12 c1(C(N2CCCC(NC(C3CN(C4CCOC4)C3)=O)C2)=O)ccc([N+](=O)[O-])s1 CC1(C)CCC(NC(c2cc(N)ccn2)=O)C(CNC(c2csnn2)=O)C1 CCC(C)(COC)C(=O)N1CCCOC(CCNC(C2(CCN(C)C)CC2)=O)C1 c1(SCC(N2CC(NC(C3C(OC)CC3)=O)(CO)C2)=O)nccc2ccccc12 C1(N(C(=O)CCC(=O)NC2CC2)C)CCC(C)(NC(=O)C#CC2CC2)CC1 C(=O)(C(C)(C)COCC(F)F)NC1(CC=C)CN(C(=O)C(O)CCSC)C1 C1(NC(CC2C(CC)C2)=O)CN(C(c2cc(C)nn2C(F)F)=O)CC12CC2 N1(C(CN(S(C)(=O)=O)C)=O)CC(OC)CC(NC(c2cccnc2C2CC2)=O)C1 O=C(CCC(=O)NCCC1CN(C(c2coc(O)n2)=O)CCO1)c1cccnc1 N1(C(C(CCN(C)C)O)=O)CCC(O)(CNC(=O)C=C(Cl)Cl)CC1 Cn1ccc(=O)c(C(=O)NCCCC2CCCN2C(c2ncc(F)s2)=O)c1 C(=O)(CC1c2ccccc2C(=O)N1C)NCC(C)NC(c1ccc(Cl)c(O)c1)=O N1(C(Cc2cc(OC)ncc2)=O)CCOCC(NC(=O)C(F)C(F)(F)F)C1 C12(C(N3CC(CC=C)C3)=O)CC(CCO1)N(C(=O)C(C1CCC1)OCC)C2 O=C(CC(F)(F)C(F)(F)Br)NCCN(C1CC1)Cc1cccc2ccncc12 c1(NC(c2ccccc2I)=O)ccc(N=c2ccn3nccc3[nH]2)cn1 C1(C(N2C3C(NC(=O)CC4COC(=O)C4)C(C3)C2)=O)CCC(C2CCCO2)O1 C1(COC)CCCCN1C(C1C=CCN(C(C)Cc2ccccc2)C1)=O CCCC(C)(C)CC(=O)NCC1CCC(NC(=O)CNC(c2cscn2)=O)C1 N1(C(c2nnn(CC)c2C)=O)CCN(C(C2CC23CC3)=O)C(CO)C1 N1(C(C(CCC)C(C)C)=O)CCC2(C=C(C(=O)N3CCCOCC3)C2)C1 C12(C(=O)NCC(c3cncnc3)C)C(NC(c3cccnc3O)=O)C3CC1C2C3 C(CNC(c1ccc(C2CNC(=O)C2)cc1)=O)(C(C)(C)C)NC(C=CCCC)=O C1(N(C)C)CN(C(C2(F)CN(C(c3cc(CO)on3)=O)C2)=O)CC12CC2 Cc1cc(C)c(C(N2CCN(C(=O)C3=CCOC3)C(C(C)C)C2)=O)c(S)n1 c1(CC)occc1C(=O)NC(CO)C(=O)NC(COC)CCO C(=O)(C(O)CCN(C)C)NC1(C(N(CCCC(=O)OC)C)=O)CCCC1 CC(C(=O)OCC1CCC(c2ccccc2)CC1)S(=O)(=O)Cc1cccc(Br)c1 c1(C(=O)NCC2N(C(c3c(C)ncs3)=O)CC(O)C2O)cncc2ccccc12 Cc1ccc(CCC(N2CCOCC2CNC(=O)C(C)CC2CCC2)=O)cc1 c1(C(=O)NCC(CNC(c2c(F)ccc(CC)c2)=O)O)ccc(OC)c(F)c1F Cc1[nH]nc(-c2nc(CS(C)(=O)=O)nn2-c2ccnc(F)c2)c1C CCC(C)CC(=O)C(=O)N1CC(O)(CNC(C2CN(C)C(=O)N2)=O)C1 N1(C(c2c(CC=C)cccc2)=O)CCN(C)C(C(=O)NC(C2CSC2)C)C1 C(C(CC(C)C)C(=O)N1C(C)C2CC1C2NC(c1nc(OC)c(C)s1)=O)OC Cc1ccc(C(=O)NCC(C)CN(C)C(c2nc(Cl)sc2C)=O)c(C)c1 N1(C(c2ccc(F)c(OC)c2F)=O)CCc2c(C(N3CC4CC4C3)=O)csc2C1 N1(C(C2C(C)(C)COC2)=O)CC(C(N2CC3(CC(O)C3)C2)=O)C(C)(C)C1 C=CCN=c1[nH]cc(C(N2CC(CCO)(NC(c3cnc(O)cc3C)=O)C2)=O)s1 Cc1ncnc(C)c1C(N1CCC(C(=O)N(CC(C)(C)O)C)C1)=O N1(CC(=O)N)CCCCC1=O.C1(O)(CNC(CN(c2ccccc2)C)=O)CN(C(N)=O)C1 CCC(CC1CCCC1)C(=O)N1CCC(F)(CNC(c2ncccc2CO)=O)C1 C1(C(=O)NCCOC(C)(C)CNC(=O)C=Cc2cscn2)(OC)CCOC1 Cc1c(NC(C(C)(C)C)c2nnnn2C)cccc1Br c1(C(=O)NC2CC(C(=O)NC(CSC)C)C2)ncc2ccccn12 c1(C(N(C(CNC(=O)C(O)CC(C)(C)C)C2CC2)C)=O)cc2cc(Cl)ccc2s1 S(=O)(=O)(c1ccc(OCC(N)=O)cc1)NCC1CCC(N(C)C)CC1 N1(C(C(CC(=C)C)C)=O)CCC(C2CCN(C(=O)C(C)Cc3cnco3)CC2)C1 c1(-c2cn(CCC(=O)NCc3nnnn3C3CC3)nn2)cnccc1Cl c1(C(=O)NCC2C(NC(C(CC)NC(C)=O)=O)CC2)ccc(C)cc1N n1(CC)nc(C(N2CCOC(C(C)NC(c3ccc(C(N)=O)s3)=O)C2)=O)cc1C C(=O)(C(CO)C(F)(F)F)NC(CCCC)CNC(C1(C)CC2(CC(=O)C2)C1)=O c1(N2CC(O)(CCNC(c3cc(C)n(C(C)C)n3)=O)C2)ccnc2ncnn12 c1(C(=O)NC2CCN(C(C3(C(=O)NC4CC4)CCC3)=O)CC2)cc(=O)c(Br)c[nH]1 C1(NC(c2cnc(CC)s2)=O)CN(C(C2(C#N)CCC2)=O)CC1SC N1(C(c2cnnc(O)c2)=O)CC2C=CC2C1CO C1(COC)CC(CNC(C2CC2C(C)(F)F)=O)N(C(=O)CS(C)(=O)=O)C1 C(CCF)(C(=O)Nn1nnc(C)c1C)C1C(C=CC)CN(C(=O)CCC2CC2)C1 Cn1nc(C(N2CCC(O)(CNC(c3cc4occc4[nH]3)=O)CC2)=O)c(Cl)c1Cl c1(C(N2C3C(N(C(c4cnc(CC)[nH]4)=O)C)CC(C3)C2)=O)nccn2ccnc12 CC(c1ccco1)=CC(=O)NC(Cc1cn(C2CCCN(C)C2)nn1)C(=O)O CCC(CCC(=O)NCCC1(NC(=O)C=Cc2cnn(C)c2)CCC1)OC CC(CC(C)(C)C)NC(C1CCC(C(C)(C)O)CC1)=O C(c1ccccc1)=C.C1(C)CCCNC(=O)C=CC=CCC(=O)N1.CC=C Cc1cc(C(N2CC(CC(F)C(=O)N(C3CC3)Cc3ccco3)C2)=O)oc1C C1(OC2(C(=O)OCC)CC=CC2)CCC(NC(=O)COc2ccccc2)CC1 c1(C(=O)NC(CC(=O)N2CC=C(C)C2)COC)cc2ccccn2c1 c1(N2CCCC(C)(CNC(C(CC)(C)CC)=O)C2)nc(C)nc(O)c1C N1(C(C(C(C)O)NC(C(C)c2ccsc2)=O)=O)CC2(CCCCCC2)C1 CC1CN(Cc2cccc(NC3CCCC3NC(=O)N(C)C)c2)C(C)CO1 CN1CCC(C(=O)NCC2CCN(C(=O)CC(C)(C)C3CC3)C2)CC1 c1(CC)cc(C(=O)NCC(C2CCOC2)NC(=O)CCc2cnccn2)n(C)n1 C(=O)(CCCC(=O)NCC1CC(F)(F)CN1C(c1cc(C)sc1C)=O)NCC CCC(C)CC(C)C(=O)NC(CC(C)(C)C)C(=O)N1CCC(n2cncn2)C1 C(c1c(Cl)nc2ccccn12)=CC(=O)NCCNC(C(C)(C)NS(C)(=O)=O)=O CC1C(NC(c2cccs2)=O)CCCN1C(=O)Cc1cc(C(F)F)no1 Cc1ccc(Br)c(CC(c2ccccc2)O)c1F C=CC1(C(=O)N(C)CCC2CCCC2)CCN(C(=O)C(C)CC=CCC)CC1 C1(NC(CC2(C)CCCCC2)=O)C2CC1CN(C(C1CCC(F)(F)C1)=O)C2 CC1(C)CC(C(N2CC(NC(=O)CN3CSCC3=O)C2)=O)CCO1 C1(C2CCOCC2)(C(=O)NCC2(C)CCN(C(c3ccsc3Cl)=O)C2)CC1 S(=O)(=O)(c1ccc(=NCc2ccc[nH]2)[nH]c1)NCCn1c(C)nnc1 C1(C(=O)NC2CC(C(C)NC(=O)C(O)c3ccsc3)C2)(OC)CCSC1 Cc1cccnc1CCC(=O)NC1CN(C(=O)CCCCNC(N)=O)CC1C c1(C(N2C(C(C)NC(C(C)C)=O)CCC2)=O)cc([N+](=O)[O-])c[nH]1 c1(N2C(NC(C(CC)OC3CCC(NCC)CC3)=O)C(C)CC2)nnccc1C#N C1(CNC(C2CC2C2CC2)=O)CCCCN1C(=O)CCC=CBr c1(C(N(C(C)CNC(C2CC2C(=O)OC)=O)CC)=O)cnc(C(C)(C)C)nc1.COC CN1CCN(C(C2CN(C(C3(C(=O)N(C)C)CC3)=O)CC23CC3)=O)CC(O)C1 C#CC1CCC(C(=O)NC2CCN(C(=O)CCc3cccc(O)n3)C2(C)C)CC1 C1(C(=O)NCCC2CC(C(=O)NCC(C(=O)OC)(F)F)C2)CC2C=CC1CC2 c1(OC)cccc(OC)c1CN1CC2CN(C(C)=O)CC12.C1(C(=O)O)CCSCC1 CCC(CCC(=O)NCC(C)(O)C1CCCC1)NC(c1nnn(C)c1C)=O N(C(=NCc1ccc(C)o1)NC1CC12CC2)C(C#C)C(C)C c1(CC(=O)Nc2cc(CC)no2)cc(OC)c(-c2ccc(CC(=O)O)cc2)cn1 N1(C(C(COCC)(C)C)=O)CCC(C2CC2)C1CNC(=O)CCc1cnoc1 N1(C(Cc2c(C)n[nH]c2)=O)CC(C(=O)NCCc2cnnn2C)C(F)(F)C1 C(=O)(C1=NOC2(CCN(Cc3ccncc3)C2)C1)NC1CCN(C(C)C)CC1 N=c1[nH]ccn2ncc(C(N3CC(CNC(c4ccnc(C(N)=O)c4)=O)C3)=O)c12 c1(C(=O)NC(C)CC(=O)NCC2C=CCCC2)cnn2cccc2c1 N1(C(C(CC=C)N(C)C)=O)CC2(CCCC2NC(c2ccc(O)c(N)n2)=O)C1 CC1COCC(CC(N2CCC(CC(=O)N(C3CCCCC3C)C)CC2)=O)O1 CCCC(CC)C(=O)NCC(C)N(C(C1CC(n2cccn2)C1)=O)CC C1(CNC(CC2CCC(C)C2)=O)CC2(CCN(C(C3CC4(CCC4)C3)=O)C2)CO1 N1(C(C2CCC(C)(C)OC2)=O)CC2(CCN(C(c3cc(CCO)on3)=O)C2)C1 c1(C(=O)NCC2(NC(=O)C#CC3(C)CC3)C(C)CCCC2)ccc2nsnc2c1 c1(OC)ccc(C(N2C3CCC2C(CNC(=O)C(C(C)O)N(C)C)C3)=O)cc1F C(C1CN(C(=O)C=C(C)c2ccco2)CC1C(=O)NC(C)C(=O)NC1CC1)=CC C(CNC(=O)C(C)(C)C)(CC(C)C)NC(C1(CCOC)CCC1)=O.C1(=O)CN1 c1(C(=O)NCC2N(C(CC=C(C)C)=O)CC(F)(F)C2)c(C)cc(=O)oc1C C(=O)(C(C)C1=CCCC1)NCC(C)N(C(c1c(C#C)c[nH]n1)=O)C N1(C(C2(COC)N(C(C(CC)SC)=O)CC=C2)=O)CCOC(C)(C)C1C N1(C(C(CC)NC(C)=O)=O)CCOCC(NC(=O)CCC2CC2Br)C1 CC(CN=c1nc2c(cnn2C)c(NCCNCCS(=O)(=O)N(C)C)[nH]1)S(C)=O CC(O)CCCCCC(=O)NC1CC2(C1)CN(C(=O)C(C)(Cl)Cl)C2 N1(C(C(C)C2CCCCC2)C(=O)Nc2ccccc2)CCCC2(CNC(=O)O2)C1 C#Cc1c[nH]nc1C(=O)NCCCCN(C(=O)CCCNC(=O)C1CC1)C N1(C(C)=O)CCCC(O)(CC(=O)NCC(C)(C)NCCc2nccc(C)n2)C1 CCCCCC(C)CC(=O)NCCOCCOCCNC(c1nocc1CC)=O c1(CC(N2C(COC)(CNC(=O)COC(C)C)CCC2)=O)cnn2ccccc12 N1(C(CC=C)=O)CC2(C1)OC1(C(=O)O)CC2(NC(c2ccc(CSC)o2)=O)C1 c1(C(N)=O)ccc(C(=O)NC(c2ccc(Br)cn2)C(F)(F)F)nc1 c1(C(=O)NC(CN(C(c2sc(OC)nc2Cl)=O)CC)C)cc(S(C)(=O)=O)c(C)o1 C(=O)(CN(C)N1CCCc2c1nc(N(C)C(C)C)n2C)OCC c1(C(=O)NC(C(C)NC(=O)C=Cc2ccc(O)cc2)C)ccn2c1CSCC2 N1(C(C2CN(CCOC)C(=O)CC2)=O)CC(NC(=O)CSC(=N)N)CC2(CC2)C1 Cc1cccc(C(=O)NC2CCC(N(C(=O)Cn3cccc3)C)C2)c1F CCCCCCC(C)C(=O)NS(=O)(=O)CC(=O)OC.C12CCC(CO1)NC2=O Cc1[nH]nc2ncc(C(=O)NCCCC(C)NC(c3cc(Cl)c(Cl)n3C)=O)cc12 C1(C(N2CCC(C(C(=O)N(C(COC)C)C)C)C2)=O)CCCSC1C c1(C(CC)N(C(=O)NCC2CCCCS2)CC)cccc(C)c1 C1(C(N2CC3CC(C2)N3C(=O)CCc2cncs2)=O)COC2(CCC2)C1 C1(C)(CC)CN(C(C2(CC)CCN(C(c3cc(OC)nn3C)=O)C2)=O)CCO1 Cc1nc(C(F)(F)F)c(NC(=O)CC2CN(C(=O)C(=O)c3ccco3)C2)s1 C(=O)(C#CC1(C)CC1)NC(C)CN(C)C(C1(c2cccs2)CCCCC1)=O CCC(CC(=O)N1CC2C(CNC(C3C4CC5C(C4)C35)=O)C2C1)CC(C)C c1(NCc2ccc(C)o2)nc2ccccc2nc1NCC1OCCc2sccc21 C12CN(CCO1)C2=O.C1(OC2CN(C(CCn3ncc(C)c3)=O)C2)CCCC12CC2 C(c1ccc[nH]1)=CC(=O)N(CCCOCCN(C(C1N(CC)CC1)=O)C)C C(=O)(CCCCCC1CC1)NCCC(C)(C)NC(C1(C)CCCNS1(=O)=O)=O C#CCC(C(=O)N(CCNC(C1(CCF)CC1)=O)CC1CC1)C1CC1 N1(C(C2(NC(CCCCCC)=O)CC2)=O)CCCN(COC)C(=O)C1 N1(C(c2c(C)onc2)=O)CCC2(CCCN(C(C3CSCCS3)=O)C2)C1 C1(C(N2CC(COC)(CNC(=O)CN3CC4CC4C3)C2)=O)CCCS(=O)(=O)C1 C12(C(N(C)CC3CCCCO3)=O)COCC1CN(C(c1ccccc1O)=O)C2 C(=O)(CC(F)(F)C(F)(F)Br)N1C(COC(C)(C)C)CCCC1 C1(C)(C(=O)NCC2CC(C(=O)NCC3(COC)CC3)C2)CCCNC1=O N1(C(c2scc(CNC(c3ccc(C)nc3O)=O)c2)=O)CCc2c[nH]nc2C1 N1(C(CCC(C)=O)=O)CC(=O)NCC1C(=O)NCC(O)C(F)(F)F Cc1nc(CCC(=O)NC(C)C(CO)NC(C2COC(=O)O2)=O)[nH]c1C Cc1cc(C(N2CCC(C(F)C(=O)Nc3cnccc3Cl)C2)=O)ncc1CO.CO S(=O)(=O)(c1c[nH]ccc1=NCC(O)Cn1ccnn1)NCC(C)F C(=O)(C1CNC(=O)c2ccnn21)NCCCCC1CN(C(CCSC)=O)C1 c1(C(=O)Oc2n(CCC)ncc2)ncc(Cl)c(SCC(=O)OC)n1 c1(C(N2CCN(C)CC2CNC(=O)C(F)CC2CCC2)=O)c2c(nn1C)CCC2 N1(C(C(N2CCC(O)CC2)C)=O)CCC(C)C(CNC(c2nccnc2N)=O)C1 N1(C(C2(C)CCC2)=O)CCN(CC2CCCN(C(C3(CC#N)COC3)=O)C2)CC1 Cc1nn(C)c2c1C(NC(=O)Cc1ccc(Br)c(C#N)c1)CCN2 c1(C(C)C)nc(=NCC2C3CN(C(C4(C)CCCN(C)C4)=O)CC23)s[nH]1 Cc1cn2cc(CC(=O)NC3(CF)CCN(C(=O)CC(=O)NC4CC4)C3)nc2s1 C(CCCC(=O)NCCn1cnc(C(=O)NCC(c2ncn(C)n2)O)c1)OC Cc1ncc(Br)c(N2CCC(O)C2C(=O)NC2CC(O)C2)n1 c1(C(=O)NCc2cc(C(=O)NCc3cc(C)no3)sc2)c[nH]c2nccc-2c1 C1(CNC(C(C)NC(CC)(C)C)=O)(NC(C2COC(=O)C2)=O)CC(F)(F)C1 c1(C(=O)NCCC(=C)CNC(=O)CSc2nncn2C(C)C)cnc(O)cc1O O=C(CCCCN1CCOC1=O)NCCCNC(=O)CCC1CC1CC1CC1 C1(C(C)NC(c2cc(C(F)F)no2)=O)CN(C(C2CCS(=O)(=O)C2)=O)CCO1 N1(C(C(CC=CC)CC)=O)CCCC(C)(C)C1CNC(=O)CNC(C)=O C1(CSc2nc(C(C)(C)C)cs2)CCCC(C#N)C1.C1(=O)CO1 C(=O)(C#CC(C)(C)C)N(C1(C(N2CC(C#C)C2)=O)CC1)C Cc1ccc(CC(N2CCCC(C(C)NC(c3cscn3)=O)C2)=O)c(Cl)c1 C(=O)(C(CN=[N+]=[N-])NC(c1cocc1C)=O)N1CC(COC)OCC1 CC(C)CCCC(=O)NC1CCCCN(C(=O)CC(C(F)F)n2cccn2)C1 CC1C(NC(c2cncc(Br)c2)=O)CCN1C(=O)COC1CC=CC1 N1(C(c2c(C)nsc2N)=O)CCC2(CCC(NC(C3(C(N)=O)CC3)=O)C2)CC1 C1(NC(=O)NCCc2ccccn2)COC2(CCNC2)C1 c1(C(=O)NC2C(C)CN(C(c3cocn3)=O)CC2)ccc([N+](=O)[O-])c(OC(F)F)c1 N1(C(CC(C)SC)=O)CCC(N(C(=O)C2=CCCS2)CC2CCCO2)CC1 CN=c1nc(C(=O)NC2CC(O)CN(C(c3ccc(C4CC4)s3)=O)C2)cc(C)[nH]1 C1(NC(C2CC(CCC)C2)=O)CCCC(NC(=O)CSc2ccccc2O)C1 c1(C(=O)NCCCC(C)NC(Cc2c(C)ccnc2)=O)ccc2c(O)n[nH]c2c1 C1(NC(C2CC(CC)OCC2)=O)CC2(C1)CC(NC(=O)C(F)(F)C(F)F)C2 Cc1ncc2n1CC(C(N1CCCCC(NC(=O)CCn3cccn3)C1)=O)CC2 C1(CC(=O)NCC2CC(C(N(CC)CC3CCCOC3)=O)C2)CCCCN1C N1(C(CC2CCN(C)C2=O)=O)CCC(C(N2CC3CCC(C2)N3C)=O)C(C)(C)C1 C1(NC(C(C2CN(C(c3ccncc3F)=O)C2)OC)=O)CC2CC1CC2(C)O O=C(CCCCCO)N1CCC(C2N(C(c3ccc(O)nn3)=O)CC2(F)F)CC1 C(=O)(C#CC(C)(C)O)NCC1CC1.CC1C(C)C(=O)N1 N=c1ccc(C(=O)NCCC2(NC(c3cn(C)nc3C(F)F)=O)CC2)c[nH]1 C(=O)(CCCS(C)(=O)=O)N1C(C)CCC(CNC(=O)CC2CCCCCC2)C1 Cc1ccc(O)cc1C(=O)N(C1(C(=O)NCC(O)C(C)(C)C)CCC1)C1CC1 C1(NC(c2c(C)nns2)=O)COCCN(C(C23CC(CO)(C2)OC3C)=O)C1 C1(C)(CN(C(C(C)OCCOC)=O)C)CCCC1NC(c1cocn1)=O C(C(C)(C)C#CC(=O)N1CC(N(C)CCO)C1)NC(C1C(C)CCOC1)=O CCC(C)C(=O)NNC(=O)NCCc1ccc(C)cc1F C12(C(=O)NC3CN(C(CC(C)n4cccn4)=O)C3)CCC(C1)C(C)(C)O2 C1(F)(CNC(C2C(C(C)(F)F)C2)=O)CCC(NC(c2csc(CO)n2)=O)C1 Cc1noc2cc(C(=O)NC3(c4ccc(F)c(F)c4)COC3)ccc12 c1(C(=O)N(CCCN(S(CC)(=O)=O)C)C)cccc(NC(=O)C(F)Cl)c1 C1(CNC(C(C)SCC)=O)(CNC(c2cocn2)=O)CCCCC1 C1(C(N2CCC(O)(CNC(C3CSCCS3)=O)CC2)=O)CCCC2CCCN12 Cc1c(Br)sc(C(=O)OCCC2CC2(Cl)Cl)c1Br Cc1nc(N2CC(C)(NC(c3cc(CO)[nH]n3)=O)C2)ncc1Cl C(CN=c1[nH]c(=NCC2OCCO2)c2[nH]ccc2[nH]1)C1CC(C)OC(C)C1 c1(C(N2C(C3CCN(C(c4cnns4)=O)C3)CCCC2)=O)ccc(Cl)c(F)c1F N1(C(CC(C=C)CC)=O)CCC2(CC1)CC2C(=O)NCC1(C2CC2)CCC1 Cc1c(C(N2CCC(NC(=O)C(F)OC(F)(F)F)C(C)(C)C2)=O)cc(C(C)C)n1C CC1COCCN(C(C2CN(C(c3c[nH]c(=S)cn3)=O)CC2(C)C)=O)C1 N1(C(C(CCCCC)=O)=O)CCC2(CC1)CC(CNC(=O)CC(C)OC)C2 Cc1cc(C(N2CCCCC2CNC(c2nc(C)nn2C)=O)=O)c2c(c1)CCO2 C1(CC)CN(C(=O)COc2cc(C)on2)CCC1NC(c1cn[nH]c1)=O C#CC1(C(N2CC(OC)C(C)C2)=O)CN(C(C2CCCCO2)=O)C1 C(C1c2ccsc2CCN1C(=O)C=CC1(C)COC1)NC(Cc1scc(C)c1)=O C(=O)(CN=S(C)(C)=O)N(CCCCN(C(CCC(=O)OC)=O)C)C CCCCC(C)C(C)(c1nnnn1CC)NCc1ccc(Br)s1 C1(C(N2CCN(C(CC(OCC)OC)=O)CC2C2CC2)=O)CCc2nccn2C1 c1(CC)cn2c(n1)CCC(C(=O)NCCCCN(C)C(c1cnc(S)n1C)=O)C2 Cc1nn(C)c2ccc(C(=O)NCCN(C(=O)C(O)c3cnc[nH]3)C3CC3)cc12 Cc1ccc(Cl)c2[nH]c(CNC(c3ccccc3OC(F)F)C)cc12 c1(C(=O)NCCC(C)N(C(COCC=C)=O)C)cc(Br)cc(F)c1F C1(C(N(C)Cc2ccc(C)cn2)=O)N(C(C2CC2(Cl)Cl)=O)CCC1(C)C c1(C(N2CCN(C(C(C)S(C)(=O)=O)=O)CC2C(F)F)=O)cccn2[nH]c(=N)nc12 Cc1ccc2c(c1)SC(C(N1CC(NC(c3[nH]cc4c3CCS4(=O)=O)=O)C1)=O)C2 C(CCN=C(NCC1CC(C2CC2)C1)NC1CCSC1C)OC(C)C C(C(C(C)(C)C)NC(C1(c2ccno2)CCC1)=O)NC(CN1CCC(C)C1)=O C1(N(C(CC(COC)COC)=O)C)CCC2CN(C(c3ccn(C)c3)=O)CC12 c1(CNC(C(c2ccccc2)C)=O)ccc2c(c1)[nH]c1ccc(Cl)cc21 c1(C(=O)NC(CC#C)C(=O)NCC(CO)C(C)(C)C)cccn2ccnc12 c1(C(=O)NCc2cc(C(=O)NC(C)C(C)n3cncn3)no2)nccnc1N Cc1ccc(OCc2ccc(-c3cncc(F)c3OC(C)C)s2)c(F)n1 c1(C(C(=O)NC)N(CC(=O)OCC)CC(C)C)cn(C(C)(C)C)nn1 N1(C(CCOCC#C)=O)CCC(NC(c2cnn(C)c2Cl)=O)C1C1CC1 N1(C(C2(CC#C)CCOC2)=O)CCC2(CCCN(C(=O)C(F)CC3CC3)C2)CC1 N1(C(c2c(C)n(C3CCOC3)nn2)=O)CCCCC(NC(C2CC(C)(O)C2)=O)C1 C(=O)(CC(C(F)(F)F)NC(C1CN2CCC1C2)=O)NCCSC(C)C C12(NC(C(CNC(Cc3c(C)cccc3)=O)C)=O)CCC(C1)OC2C c1(NC(C2CC3(CC3)CN2C(C2C=CCCC2)=O)=O)ccc2c(c1)OCC2 N1(C(C2CCN(C(CC)=O)C2)=O)CCCC(CCNC(c2cc(O)no2)=O)C1 N1(C(c2cc(OC)nc(OC)c2)=O)CCCN(C(=O)C(C)NC(C)=O)C(C)C1 C(N=c1nc(C)nc2[nH][nH]cc1-2)C1(NC(C)=O)CCCC1.C12CCN(CC1)C2=O Nc1ccc(C(N2CC(NC(c3cc4ccsc4s3)=O)C(O)C2)=O)cc1Cl Cc1cc(=NCC2(CCNc3nccc4ncnn34)CC2)[nH]c(C(C)(C)C)n1 c1(N2CC3CC(NC(c4cncc(OC)n4)=O)C3C2)ccc(C#N)c(C)n1 C1(C(=O)NC(C)CN2CCCC2)CC2CCC(C1)N2C(=O)C(F)F C1(CCNC(COCCCCC)=O)CN(C(=O)Cc2nnc(CC)o2)CC(C)O1 CC1(NC(=O)C(O)CCl)CCN(C(=O)NC2(c3cccc(Cl)c3)CC2)C1 Cc1c(C(=O)N(CCCCCC(=O)NCC(c2ccnn2C)O)C)[nH]ccc1=O CCC(CC)CC(=O)N1CCN(C(c2cnn(C)c2Cl)=O)C(CCO)C1 C1(NC(C(C)(CO)NC(C)=O)=O)CC2CC1N(C(C1CCC(C)CC1)=O)C2 C1(NC(=O)CCC2CCCN2C(c2coc(C(F)F)c2)=O)CCCC(CO)C1 C(C)(C(=O)N1CCC1C(=O)NCCCOCCCO)=C(C)C.C(C)(C)O N1(C(C=CCN(C)CC)=O)CCC2(CC1)CN(C(=O)C(O)C1CCCC1)C2 N1(C(CC2(C)CCCC2)=O)C2CC1CN(C(=O)Cc1sccc1Cl)C2 c1(C(=O)NC2(C)CC(NC(C(C)C(C)(F)F)=O)C2)cnn2cccnc12 Nc1c(F)ccc(F)c1C(=O)NCC1CC1NC(C1(C(F)(F)F)CCCCC1)=O C1(CC)CN(C(c2ccc(Cl)cc2)=O)CCC1NC(=O)Cc1cn(CC)nn1 C=CC(C)(CC)C(=O)N1CCCOC(CNC(C2CCCC2)=O)C1 Cc1cc(C(=O)NC2CC2CNC(=O)CC2CC3(CC3)C2)c(C)cc1Cl C(=O)(C(N)CCS(=O)(=O)N1CCCCCC1CC(C)C)OC C=CCC(CC=C)C(=O)N1CCCC(N(CCO)C(c2ccc(C)nc2C)=O)C1 n1(CC)nccc1C=CC(=O)N(C1CN(C(C2CC(CF)C2)=O)CC1O)C CC1CN(Cc2ccccc2-c2nn[nH]n2)CC(C)N1C(=O)C1CC1 C1(C(N2CC(C(=O)NCC)C2)=O)N(C(c2cc(COC)no2)=O)CCC1(C)C C1(CC(C)NC(COCCCC)=O)CC2CCC(C1)N2C(c1ccc(O)cc1)=O C#Cc1ccc(F)cc1C(=O)NC1CC(C)N(C(C2OCCN(C)C2=O)=O)C1 CCCCCCC(C)C(=O)N1CCC(O)(CCNC(C2(CC3CC3)CC2)=O)C1 C1(C(=O)NC2CCCC(NC(C3CCCO3)=O)C2)C2CC(F)(F)CC12 CC(C)(CCNC(=O)COc1ccsn1)NC(=O)Cn1ccc(C2CC2)n1 N1(C(=O)COC2CCCC2)CC2CCC(C1)N2C(c1ncc2[nH]ncc2n1)=O CN1CCN(C(c2cc(F)cc(F)c2)=O)CC1CNC(=O)CCC1CC1 C(=O)(C(CCC)CC(C)C)NC1CC(CCC(=O)NCCCC(C=C)(C)C)C1 c1(CC(=O)NC2C(NC(C3N(C)CCOC3)=O)CCC2)cc(F)ccc1O Cc1ccc(C(O)C(=O)NC2COCC2NC(=O)CCOCC(F)(F)F)cc1 C1(N(c2ncc3[nH]ccc3n2)C(c2nc[nH]n2)=O)CCCC12CCNCC2 c1(OC)c(C(=O)NCC2(CNC(C3(C)CC3C)=O)CC23CCC3)ccc(Cl)c1C C(=O)(CCC(=O)C(C)(C)C)NCC1C(C(N2CCC(C(C)CO)CC2)=O)CCC1 c1(NC(=O)NCc2nc(CC)on2)cccc2c1C(C)CC2(C)C C1(CNC(c2ccoc2Cl)=O)CN(C(c2sccc2F)=O)CC2(CCC2)O1 C1(C(=O)NCCCCC(C)NC(C2CC3CCC2CC3)=O)CCCCCN1C [N-]=[N+]=Nc1ccc(C(=O)NC2COCCN(C(C3C=CCS3)=O)C2)cc1 CC1CCC(NC(C2CC23CC3)=O)CN1C(=O)C1=COCCC1 C1(NC(Cn2ccc(C)cc2=O)=O)CCN(C(C2(O)CC(C)C2)=O)CC12CCC2 c1(C(N2CC(NC(c3cc(Cl)ncc3F)=O)(CO)C2)=O)ccc2cnoc2c1 C1(CNC(C2C(C)C(=O)C2)=O)(NC(=O)C(=O)N(C)C)CCCCCC1 CC(C)(C)S(=O)(=O)CC(=O)NCC1CCCN1C(=O)CCc1cncs1 C(N=c1nc2c(Br)csc2c[nH]1)C1C(NC(=O)CC(F)F)CCC1 N1(C(C2C(C3CN(C(C4CCSCC4)=O)C3)C2)=O)CC2CCC1C(O)C2O c1(C(N2CCCCC(NC(C(CC)CC)=O)C2)=O)[nH]c2ccccc2c1C#N N1(C(Cc2c(C)cc(F)cc2)=O)C2CCC1CN(C(c1ccc(Cl)o1)=O)CC2 C1(C)(CC)CCC(C(=O)NCCOCC(C2CCCCC2)=O)O1.C(CC1CC1)O CC(C(=O)NC1CN(C(c2cc(N)ccc2F)=O)CC1C(F)(F)F)C1=CCCC1 N#Cc1cc(C(=O)NCC2CC2CNC(c2ccc(Cl)s2)=O)cc(F)c1F N1(C(C=CC)=O)CCN(C(c2cc(C)c(Cl)c(N)c2)=O)CCC1C C(C(C)CC(=O)N1CCC(CN(C(=O)CCc2ccc[nH]2)C)C1)OC c1(C(=O)NCC2CCC(NC(c3nncc(C)c3)=O)C2)cncc2cnccc12 CCC(CC(=O)N1CCN(C(c2cnc(C(N)=O)s2)=O)CCC1C)CC(F)(F)F C1(NC(Cc2nc(C)[nH]n2)=O)CCCN(C(=O)C(C(C)C)SC(F)(F)F)C1C C(C(=O)NC1(C(F)F)CCCC1)(C(C)C)NC(CCOCCOC)=O c1(NC(C2C(C(C)NC(C3CN(C(N)=O)C3)=O)C2)=O)ccc2c[nH]nc2n1 C1(COC)(NC(=O)CSC2CCOC2=O)CCN(C(C2CCS2(=O)=O)=O)CC1 c1(C(=O)NC2CC(NC(c3c(Cl)cc(C)c(F)c3)=O)C2)cc(F)c(F)c(F)c1F N1(C(CNC(N)=O)=O)CC2CCOC2(CNC(=O)CN2CCC(O)CC2)C1 C1(C)(C(=O)NCC(CNC(c2c(C)nc(=N)[nH]c2)=O)O)CCCCC1(F)F N1(C(C2C(CC)CCC2)=O)CC=C(CCNC(=O)C=CC2CCCCCC2)CC1 C1(NC(c2c(C)nc(O)cc2)=O)CC2CN(C(=O)C(O)C3CCC3)CC2C1 C(C(C)(C)CC(=O)NCC(O)C(C)O)NC(c1cccc(CC)n1)=O C(CNC(C1CCC(C)O1)=O)(C(C)(C)C)NC(Cn1ncc(C)c1)=O C(COC)(C(=O)NCCO)N.C(CC(=O)N(C)C)NCC(=O)OC(=O)NC C(CCC(C)(C)C(=O)NC(c1cccc(F)c1)C)NC(CCCCC=CC)=O Cc1cnc(CNC(=O)CC2CCCCN2C(=O)COc2ccon2)c(F)c1 N1(C(CSC)=O)CCC(C(=O)NC2C3CCC2CC3)C1C(C)C CN1CCN(c2ccc(C(=O)NC3CCN(S(=O)(=O)CC#N)CC3)cc2)CC1 CC1(C)C(=O)NCC1NC(=O)CC1CCCCC1NC(C1(C)CCCO1)=O C1(CNC(C2C(CCC)C2)=O)CCCC2CN(C(C3CCCCC3C)=O)CC12 c1(CN(C(C)(CO)C2CCC2)C)ccc(S(=O)(=O)N2CC3CC3(CO)C2)cc1Cl C(CC(=O)Nc1cnncc1OCC)(C(F)F)NC(C(C(C)C)OCC)=O Nc1nccnc1C(=O)NCCCCNC(=O)CCc1ccc(Cl)nc1 c1(-n2c(C)nnn2)ccc(C(=O)NC2CC(F)(CNC(c3cccs3)=O)C2)cc1 N1(C(c2nn(C)c(C(F)(F)F)c2)=O)CCCN(C(C2CCC3CC23)=O)CCC1 C=CC1(CC(=O)N(C)CC2CCCN(C(=O)C(O)C(C)(C)C)C2)CCCCC1 c1(C(N2CCCN(C(=O)Cc3cscn3)C(CO)C2)=O)ccc(F)c2occc12 c1(CN2C(C(=O)Nc3ncccc3F)CNCC2)c[nH]c2ccc(Br)cc12 C1(NC(=O)C(C)(C)Cl)CCC(C(N2CC(CC(C)(C)C)C2)=O)C1 Cc1cc(Br)c(C)c2sc(C(N3CCCC(C)(N(C)C)C3)=O)nc12 CC1(C)C2CN(Cc3cncc(O)c3)C(C(N3CCCCC3)=O)C12 S(=O)(=O)(CCC(=O)NC(C)CCNC(=O)COc1ncccc1C#N)NC C1(OC)CN(C(C)C)CC1NC(c1cn(C(F)(F)F)nc1C)=O C#Cc1cnc(C(=O)NC(C)(C(C)Sc2ccccc2)c2ccccc2)c(C)c1 CC(C)=C=CC(=O)NCC1CC(C(N2CCC(CO)(CO)C2)=O)C1 CN=C(NCCc1ccccc1O)N1CCC(CN2CCOC2=O)C1 N1(C(c2c(CC)non2)=O)C(C(=O)NCC2(CSC)CC=CC2)CCC1C1CC1 N1(C(CCc2n(C)ccn2)=O)C2CCC(C(N3CC=C(CO)CC3)=O)C1CC2 CP(C)(=O)c1ccc(C(=O)NCC23CC(CO2)N(c2ncc4ccnc-4[nH]2)C3)o1 N1(C(c2ccc(C(C)=O)s2)=O)CCCC(CCC(=O)NC(c2ccn(C)n2)C)C1 C=CC(C)(C)CCNC(c1ccc(CNC(C2(C)COC2)=O)o1)=O C12(NC(Cc3ccc(C)o3)=O)CCCC1CN(C(=O)Cn1ccsc1=N)C2 C12CCC3(CC(C3)CC3CCCN(C3)C1=O)O2.C(=O)(CCCn1ccnn1)N(C)C c1(C(N2CC(C)N(C(c3cnc(C(C)(C)C)[nH]3)=O)CC2)=O)cccc2[nH]ncc12 c1(CCC(=O)NCC(C)CN(C)C(C2CC3(CC3)CO2)=O)nncnc1O C(=O)(C(C(C)(C)C)n1ccnn1)N1CC(NC(C2(C#C)CC2)=O)C(COC)C1 c1(C(N2CC(CC)(NC(=O)CC(C)(C)OC)C2)=O)cc(C)nnc1O c1(C=O)cccc(O)c1.n1(CC)cc(NC(c2c[nH]nc2CC)=O)cn1 N1(C(c2cccc(I)c2)=O)CCC2(CCCN2C(=O)NC2CCC2)C1 C=CCCCCC(C)c1nc(C23COC(CCO2)C3)no1 C(CCC(=O)NCCN(C(c1cc(CCO)on1)=O)C1CC1)C1C(C)C1 CC(C)CCCCCC(=O)N(C(C)CNC(C1CCC(F)(F)C1)=O)C C(C(F)(F)C(C)(C)O)NC(C1CC(C)(NC(c2c(OCC)cccc2)=O)C1)=O c1(C(=O)NC2CC3CC(NC(c4cn(C)nc4)=O)C3C2)cnc2c(n1)CCCC2 c1(CC(N2C3CN(C(CCC(C)OC)=O)C(C3)C2)=O)ncn2c1COCC2 N1(C(c2cnn(CCNC(C3(F)CCOC3)=O)c2)=O)CC2CC1CS2=O c1(C(N2C(CNC(c3c(C)ccc(CC)c3)=O)C=CC2)=O)cc(O)cc(N)c1Cl n1(CC(=O)NCCNC(c2c(C)oc(C#N)c2)=O)nc(C(F)(F)F)c2c1CCC2 N1(C(C(CNC(C2CCN(CC)C2)=O)C(C)C)=O)CC(C2=NOCC2)C1 CC1(C)CCC(CNC(=O)NCCN2CCN(C3CCNC3)CC2)C1 N1(C(CCc2nc(C)c(C)o2)=O)CCC(C2CC2)(NC(=O)CSc2cn[nH]c2)C1 c1(C(=O)NCC2(C)CCCN(C(c3cc(C)sn3)=O)C2)c[nH]c2cc(O)ccc12 C(C1=NOC2CCCC12)NC(C1N(C(c2cc(C)c(C)nc2)=O)CCC(O)C1)=O C1(C(=O)NCC2C(C)CN(C(=O)CN3CC4CC4C3)C2)COc2ccccc2O1 C1(CC(=O)OCC)(C(=O)Nc2c(C(N3CCC(CF)C3)=O)c[nH]n2)CCCC1 c1(SC)cncc(C(=O)NCC2(O)CCN(C(=O)CC3CCCO3)C2)c1 c1(CCN(C)Cc2cn(CC(N3CCC(C(C)(C)O)C3)=O)nn2)ccc(Cl)cc1 Cc1ccc(C)c(OC(C2CCC2c2ccc(C#N)cc2)=O)c1 c1(CC)nc(C)c(C(=O)NCC2(F)CCC(NC(c3nnsc3C)=O)C2)s1 n1(CC)nc(C)c(CC(=O)NCCC(C)NC(C2CCCCC2C(N)=O)=O)c1C C1(C(=O)NC(CC)C(C)CN(C)C)CC2CCC1N2C(=O)C=CC1CC1 C1(C)(NC(CSc2n(C)cnn2)=O)CCN(C(=O)C(N2CCCC2=O)F)C1 c1(CC(=O)NC2CC(NC(=O)CNC(=O)C3CC3)C23CCC3)cc2occc2s1 Cc1ccc(CC(N2CCC(NC(=O)Cc3ccc(Br)s3)C2)=O)cc1C c1(CC)cc(C(N2CSCC2C(=O)NC2(C(N)=O)CCOC2)=O)ccn1 N1(C(c2n(C)cc(C#N)c2)=O)CC2CCC(C1)N2C(C1CCOCC12CCC2)=O c1(C(=O)NCC2(NC(=O)CNC(c3cccs3)=O)CCOC2)ccc(F)c(F)c1 C1(C(N2CC(N(C(C(CC=C)NC(C)=O)=O)C)C2)=O)CC2CC1CC2=O C1(NC(c2scc(C)c2C)=O)CCN(C(=O)CN2C(=O)CN(C)C2=O)CC1C CCC(C)(C)C(O)C(=O)N1CC(C(=O)N(CCO)CC2CC2)C2(CCC2)C1 CN1C2CCC1CN(C(=O)C(c1cccnc1)NC(c1cncc(O)c1)=O)C2 Cc1cc(CCCNC(C2CCCN2C(=O)CCCNC(=O)NC(C)C)=O)no1 c1(C(=O)NC2C(CNC(c3c(C)[nH]cc3)=O)CCC2)oc2cc(Cl)ccc2c1C C1(C(N2C(C)(C)C=CC2)=O)COCCN(C(=O)COC2CCOCC2)C1 C(=O)(CCCC(C)(C)C)N1CCC(C(C)C(N2CCCC2c2ccon2)=O)CC1 C1(CNC(C=C(C)C(C)C)=O)COCCN1C(=O)C(c1ccc(N(C)C)cc1)C N1(C(C(CC(C)C)c2ccc(Cl)cc2)=O)CC(C)(C)c2ccccc21 c1(C(N2C(CO)CC(C(=O)NC3(CC=C)CCOC3)C2)=O)ccc([N+](=O)[O-])[nH]1 C(N=c1[nH]c(=NCc2nccc(O)n2)[nH]c2c1CCCC2)c1cc(C)cc(Cl)c1 c1(CNCC(COC(C)C)OCC)ccc(OC)nc1 n1(CCC(=O)N(C)CC2CCCN2C(=O)CCOC)cnc2cc(F)c(F)cc12 n1(CC(N2CC(C3(NC(C(CC)C#N)=O)CC3)C2)=O)c(C)cc2ccccc12 C(=O)(CCC(=O)C(C)(C)C)NC1CC(C(N2CC(SC)C2)=O)C1 C1(C(=O)NC2(C3CCN(C(C4(C#C)CC4)=O)C3)CC2)Cc2ccccc2C1(C)C c1(CC)nonc1C(=O)NC1CC(O)(CNC(C2CCN2S(C)(=O)=O)=O)C1 c1(NC(c2c(NCC3CCN(CC)CC3)cc(Cl)cc2)=O)ncnc2cc[nH]c12 C(=O)(C(CC(C)C)OC)N(CCCCCCNC(C1C(C(=O)OCC)C1)=O)C N1(C(CN(CCC)C)=O)CCC(N(CCOC)C(C2CCC2OC(C)=O)=O)CC1 C1(NC(c2cn(CC=C)nn2)=O)CCOC(C(=O)N(C)CCc2cccs2)C1 N1(CCN(C(C(N2C(CC)CCC2)=O)=O)C)CCN(C(=O)COC)CC1 N1(C(=O)C(F)=C2CC2)CCCC(N(C(=O)Cc2c[nH]ccc2=O)CCO)C1 C(CC(=O)NC(CNC(=O)C(CC)N1CCNC1=O)C1CCC1)(OCC)OCC c1(C(=O)NC(CNC(C(C(C)C)OC)=O)C2CCC2)ccc2oc(S)nc2c1 CC(CC(C)(C)C)C(=O)N(CCCCNC(=O)CSCC(N1CCCCC1)=O)C C1(OC)CCCC(CNC(C2C(C)CCN2C(=O)CSC(F)F)=O)C1 N1(C(CC(C)(F)F)=O)CCC(O)C(NC(=O)CCNC(C2CCCCC2)=O)C1 C1(C(=O)NC(CC2CN(C(CCC=C(C)C)=O)C2)C)CCn2cncc2C1 N1(C(C(CCC2CCC2)NC(CC(COC)(C)C)=O)=O)C2CCC1CC(=O)NC2 CN1CCCCC(C(=O)NCC=CCNC(=O)Cc2c(F)cccc2F)C1=O C1(O)(c2cn(CC(N3C(COC)CCCC3)=O)nn2)CC2CCC1C2 C1(CCC)CCCC1C(=O)NC1CC(C)(NC(=O)CC2CC3CC3C2)C1 C(=O)(C1=NNC(=O)C1)N1CC(COC)(NC(=O)COCc2cc(C)no2)C1 N1(C(c2cc(CC)ncn2)=O)CCN(C(C2CCN(C)C(=O)C2)=O)C(C2CC2)C1 Cc1nc(=NC(C)Cc2ccc3c(c2)CCO3)[nH][nH]1 C(C)(CCCCO)NC(=O)CCCSC.C(C)(C(=O)NC)SC CC(C)(CCCO)C(=O)N1CCCC2(NC(=O)COC(F)F)CC2C1 C1(CNC(c2cn(CC=C)nn2)=O)CC(C)(C)CN1C(c1csnc1Cl)=O c1(C(=O)OC)c(N2CC(NC(=O)CCCCN(C)C)CCC2C)ncnc1Cl CN1CCC(CN(C(C2CCC2NC(=O)Cc2ccc(O)nc2)=O)C2CC2)CC1=O C1(C#N)(C(=O)NCC(CNC(c2cnc(C3CC3)o2)=O)OC)CC2CCC1CC2 N(C(=NCCC1CC1)NCCC1CCCC(C)C1)C(C=C)C N1(C(=O)OC(C)(C)C)CCC(CCCCC(=O)N2CC3C(C(N)=O)C3C2)CC1 C1(CC(=O)NCCCCC(=O)OC)C2CCC(C2)N1C(C1CCC1C(C)(C)C)=O Cc1nc(C(C)C)oc1C(=O)NC1(C)CCN(C(=O)CC=Cc2ccccc2)C1 C(=O)(CC(C)(C(F)(F)F)N(C)C)NC1CCN(C(c2nc(OCC)oc2)=O)C1C Cc1occc1C1(C(=O)NC2CCCC2CNC(C2(C)COC2)=O)CC1 N1(C(c2c(OC)nccn2)=O)CC(CNC(C2CC(=O)N(C)C2)=O)OC(C)(C)C1 C1(C(=O)NC2CCOC2)CC2(CC2)CN1C(c1cnc(C(F)(F)F)s1)=O Cn1cc(S(=O)(=O)NCC(=O)NCCNC(C2(C)CCCCC2(F)F)=O)cn1 C(=O)(C1=CCCC1(C)C)NCC1CCN(C(C2C(C)(C(C)C)C2)=O)CC1 c1(NC(C(C)C)C(C)NC(c2cnnn2C(C)C)=O)ccc([N+](=O)[O-])cn1 c1(CN2C(C(N3CCOC(c4ccc(Cl)cc4)C3)=O)C=CC2)cc(Br)cnc1O CC1CCN(C(C2CCC(=O)N2C)=O)CC1NC(c1cn(CCC2CC2)nn1)=O c1(C(N(C(CC)CNC(=O)C(C)OC)C)=O)cc(OC)cc(F)c1 C1(CNC(C2(CC)CC2)=O)CCCN(C(=O)CN(c2ccccc2)CCOC)C1 c1(C(=O)NC(CNC(c2coc(Cl)c2)=O)C2CC2)cc2ncccc2[nH]1 c1(OC(c2ccc(CC)cn2)=O)ccc(Cl)cc1F.c1(N2C(=O)C2)ncc[nH]1 C1(C(=O)NCC(CCNC(=O)C=CBr)OC)CCc2nnc(O)n2C1 C1(NC(CN(CCC)C(c2cnc(C)cc2F)=O)=O)CCCC(C2CC2)C1 c1(C(=O)NCC(CO)NC(c2cnc(CC)[nH]2)=O)ncncc1OC C(=O)(C(C)C(O)C(C)CC)N1CC(C#C)(C(N2CC3CC2CS3=O)=O)C1.C1CN1 c1(OC)cccc(C(C)CC(=O)NCCN(C)C(c2c(C)csc2C)=O)c1 c1(C(=O)NCC2C(C)CCN(C(=O)C=Cc3cn[nH]c3)C2)nc2ccccn2n1 c1(CC(N2CCN(CC(C)N)CC2)=O)c(C)nn(CC(C)C)c1Cl.CO C12(C(N3C(C(C)O)CC3)=O)CCCC1CCN2C(=O)Cn1cc(C)cn1 C1(NC(c2ncn(CC)c2)=O)CC12CCN(C(=O)CCC(C)C)C2 N1(C(C(CCC)C(C)C)=O)CC=C(CC(=O)NC(CO)C2CC2)CC1 Cc1c(NC(c2ccnc(C3CCC3)c2)=O)cnn1-c1ccc(F)cc1 CCC(C)(C(=O)N(CCNC(=O)CSc1cccc(C)c1)CC1CC1)OC C(=O)(CC1=CCOCC1)N(C)C(=O)OCCOC(=O)CCC(=O)c1ccc(Cl)s1 c1(CC)ccc(OC)c(C(=O)NC2CCC(NC(C3(OC)CCOC3)=O)CC2)c1 c1(C(=O)NC2CCN(C(C=Cc3ccc(C)o3)=O)CC2O)scc2c1CCCC2 Cc1noc2cc(C(N3CCC(C(F)CNC(=O)CCF)CC3)=O)ccc12 N1(C(C(C)CC(F)(F)F)=O)CCCCC12CN(C(=O)CN1CC=CC1)C2 c1(C(N2CC3CC3(C(=O)Nc3ccncc3)C2)=O)ccnn2ccnc12 C(CCC(=O)N1CCCC1CC(=O)N(C(CC)C1CC1)C)OCC=C c1(C(N(C)CC2(NC(COCC(=O)NC)=O)CC2)=O)cccc(C(C)=O)c1 C(=O)(C(F)(F)C(F)(F)F)N1CC(CC(=O)OC)(NC(=O)C(CCC)N(C)C)C1.C=CC C1(C(=O)NC2CC(NC(CC(C)(C)F)=O)C2)COc2cc(F)ccc2C1 c1(C(C(=O)N(CC(F)F)C)NC(C(C)n2cccn2)=O)cn(C)nn1 N1(C(=O)CCC#N)CCCCC1c1cn(CCN(CCO)CCO)nn1 C1(C2CCOCC2)(C(=O)NCCCN(C(C)=O)C)CCNC1 c1(NC(C23C(NC(c4c(C)snc4)=O)C4CC2C3C4)=O)ccc2nccn2c1 Cc1cc(O)nnc1C(=O)NC1CCN(C(c2cc(F)c[nH]2)=O)C(C)C1 Cc1ncc2n1CCC(C(=O)NCC13CC(CN1C(=O)Cc1cscn1)C3)C2 C1(NC(C(CCC#C)NC(=O)Cc2cn(C)cn2)=O)C(=O)OC2CCCC12 C=CCC(CNC(=O)C(C)NC(=O)CSCNC(c1cc(OCC)no1)=O)OC c1(CC)cc(C(=O)NC2CC(C)(CNC(=O)C(C#N)CC)C2)cc(Cl)c1 C1(C(N(C(CC#C)C)C)=O)CC12CCN(C(c1ccc(O)c(F)c1)=O)CC2 c1(N2CCC(NC(N(CCCOC(C)(C)C)C)=O)C2)ccc(F)cc1F C(c1ccncc1)=C(C)C(=O)N(C1CN(C(=O)C(c2ccc(Br)o2)C)C1)C c12cc(ccn1)CNC(=O)C1(CC1)N(CC(C)C)C2=O.C1(NC(C)=O)CCC1 N1(C(c2c(OC(C)C)nccc2)=O)CC2CCC1(CNC(=O)C1CC1)CC2 N1(C(c2c(CC)nn[nH]2)=O)CCN(C(=O)C(C)O)CC1c1ccc(CC)o1 C1(C(=O)NCC2(C)CC(C)(C)C2)N(C(=O)Cc2ccc[nH]2)CCCC1(C)C C(=O)(C#CC1CCOC1)NCCCCC(C)(C)N(C)C.C(C(C(=O)N)OC)OCC c1(CC(=O)NC(C)CNC(C23COC(C2)C3)=O)cc(Cl)ccc1Br N1(C(c2n[nH]cc2[N+](=O)[O-])=O)CCC2CN(C(c3ncc(Br)cc3Cl)=O)CC2C1 N1(CCC(=O)NCC(C)(C)CNC(=O)Cc2cn[nH]c2)CCCCC1=O C=C1CCC(C(=O)NC2CCN(CCCNC(c3c(C)[nH][nH]c3=N)=O)C2)CC1 C#Cc1ccc(C(N2CCC(C)CC2C(N2CCC(COC)CC2)=O)=O)c(C)c1 C1(F)(CNC(c2nc(C(C)C)sc2)=O)CCN(C(=O)C=CC(C)(C)C)C1 C1(C(N2CCC(C(C)(C)O)C2)=O)CCn2c(nnc2Br)C1 Cn1nc(C(=O)NCCNC(C2C(c3ccccc3)C2(C)C)=O)c(Br)n1 C1(NC(Cc2c(C)ccs2)=O)CC2CCC(C1)N2C(=O)CCCc1cccnc1 C=CCCC(CC(C)C)C(=O)NCC1CCC1NC(c1cnc(N(C)C)o1)=O CCCC(CC)C(=O)NCc1cc(C(=O)N(C2CC(F)(F)C2)C)ccn1 c1(C(=O)NCc2ncn(-c3ccccc3)n2)ccc(F)c2cccnc12 C1(CC(=O)Nc2c(C)nccn2)CCCC12CN(Cc1ccc(C)c(O)n1)C2 Cc1cc(CN2CCCC2(C)C(=O)Nc2ccccc2Br)c(O)c(C)c1 N1(C(C)=O)CCC(NC(=O)CC2CN3CCC2CC3)CC1C N1(C(c2n(C)nc(Br)c2)=O)CC2CN(C(c3cc(C(C)(C)C)n[nH]3)=O)CCC12 c1(CC(=O)NCCC2(CO)CCC2)ccsc1C(=O)NC1CC(CCF)C1 c1(C(N2CC(C(=O)OC)C(C(C)C)C2)=O)cc(C)c(F)c(C)c1.c1ccc(CO)s1 c1(C(N(CC(O)CNC(=O)C2=NNC(=O)C2)C)=O)c[nH]c2cc(Br)ccc12 Cc1ccc2[nH]c(CNC(c3cccc(-n4cncn4)c3)=O)cc2c1 Cc1cc2c(o1)CC(C)(C)CC2NC(=O)N=c1cc(CCc2ccccc2)o[nH]1 c1(C(N(CC(CC)NC(=O)CCC2CCC(=O)N2)C)=O)cc(C)n(C(C)(C)C)n1 N1(C(=O)OC(C)(C)C)CCCCC(NS(=O)(=O)NC2COC2)C1 C(=O)(C1=CC2CCCCCC12)N1CCC(C(=O)NC2(CC(C)=O)CCCC2)C1 c1(OC)ccc(C(C)NC2(c3nnnn3C3CCC3)CC3CC3C2)cc1 N1(C(CN(C(=O)OCC)C)=O)CC2CC2(NC(=O)Cc2cc(C3CC3)no2)C1 C(C)(C(=O)N(C)CCN(C(C1(C)CC1Br)=O)C(C)C)OCCOC c1(N(C)Cc2ncc(Br)s2)nc(NC2COCC2F)c2ccsc2n1 c1(C(=O)NC2C(NC(c3c(OC)n(C)nc3C)=O)C2)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)NC(C(C)NC(C2CC3COCC3C2)=O)(C)C)cc2ccccn2n1 CC1=NC(C(=O)NCC(O)CNC(c2ncoc2C(F)(F)F)=O)CS1 C1(NC(c2c(C)n[nH]c2C)=O)CCCCN(Cc2nc(C(C)(C)C)no2)C1 Cc1ncccc1CCC(=O)NCC(c1ccccc1)NC(=O)Cn1cnnc1 Cc1ccc(CC(N2CCCC(C(C)C(=O)NC3CCSC3C)C2)=O)cc1 c1(COC)ncc(C(N2CCCC2CCNC(=O)CCN2CCCC2)=O)s1 c1(C(=O)NCC(C)(C2CC2)NC(c2cc(CC)nn2C)=O)c(C)nn(C)c1OC C1(C(=O)NCCSCC(=O)NC(CC)COC)CCCOC1(C)C C1(NC(C2(CN(C)C)CC2)=O)CC(C(=O)NCCN2CCCC2)CC1O C1(NC(CSCC(N)=O)=O)CC2CCC1(CNC(c1nn[nH]c1Cl)=O)C2 CC1(C)CCC2(CC1)CC2C(=O)Nc1cncc2ccccc12 C1(Cn2c(C)nc(-c3ccc(F)cc3)n2)COCC1CS(C)(=O)=O CC1(C)CC(CNC(c2cnc(O)nc2O)=O)N(C(=O)CCN2CCCCC2)C1 c1(C(N2CCC(CCc3ccccc3)C2)C)nc2c(s1)CCC2 c1(C(=O)NC(CNC(C2(CCCC)CC2)=O)CO)cc(C)n(C2CCOC2)c1C C1(N(C)C(c2ccn(C)n2)=O)CCCC2CN(C(C34CCCC3C4(F)F)=O)CC12 c1(C(N2CCOCC2CNC(C2CCCC(C)C2)=O)C)cccc2ccccc12 c1(OC(C)C(N2CCN(C(c3ccon3)=O)C(C)C2)=O)cccc2ccccc12 N1(CC)CC2CN(C(C3C=CCN3C(=O)C(c3cncnc3)C)=O)CC2C1 C(=O)(C(F)C(=O)NCc1n[nH]cc1C(=O)NCC(C1CCOC1)O)OCC Cc1cc(C)nc(N(C2CCCNCC2)C(=O)CCc2cccs2)n1 C1(NC(C2C(CC)OCC2)=O)CN(C(=O)CCC(C)SC)C2CCCCC12 N1(C(c2cc(C)cc(O)c2)=O)CC2(CCN(C(C3CC4CCCC4C3)=O)C2)C1 C1(NC(C(C)c2cccs2)=O)(CF)CCN(C(c2cc(C(C)(C)C)on2)=O)C1 C=CC(O)C(=O)NC(C1CCCCC1)C(=O)N(CCO)CCOC N1(C(CC(CC)OC)=O)CCC(CCNC(C2(Cl)CCC2)=O)CC1C c1(CN(C=O)CC(c2ccc(Cl)c(Cl)c2)O)cc(Cl)ncc1Br CC(CO)(C(F)(F)F)NC(=O)CC1CN(C(=O)CC23CC(C2)C3)C1 S(=O)(=O)(c1cc(C(=O)N(C(CNC(c2ccc(F)s2)=O)C2CC2)C)co1)NC C(=O)(C(C)(O)C(F)(F)F)N1C(C(=O)NCC(C)CC2CCC2)CC(F)C1 c1(OCCn2c(C3(C#C)CCCC3)nnc2N(C)C)cnc(Cl)cc1C N1(C(CCNC(CC(C)C)=O)=O)CCC(O)(C(=O)NCc2cncc(O)c2)CC1 Cc1cc(O)ncc1C(N1CC(C(O)C(=O)NC2C=CCCC2)C1)=O C1(NC(c2c(C)cnnc2)=O)CCSC12CN(C(=O)CN1CSCC1=O)C2 c1(C(=O)NC2CC2CNC(C2C3CCCCC23)=O)c(Cl)ccc2cccnc12 c1(NC(C(CC2CCC2)NC(=O)C=Cc2cscn2)=O)ccc(CCO)cc1 c1(C(=O)NC(CCOC)CNC(c2cnc(-c3cccs3)o2)=O)c(Cl)cnn1C c1(CC(=O)NC2C(C)CN(C(=O)C=CC3CCC3)C2)cnc2cccnn12 S(=O)(=O)(C1CC12CCCCC2)C(N1CCC(n2cc(-c3n(C)cnc3)nn2)C1)=O C1(C(N2CC(NC(CC3CCC(=C)CC3)=O)C(C)(C)C2)=O)CCCCN(C)C1=O N1(C(c2c(C(C)C)ncs2)=O)CCCC(C2(NC(=O)CC(F)(F)F)CC2)C1 c1(C(=O)NC2CCCC(CNC(C(C)(C)N(C)C)=O)C2)cc2c[nH]nc2s1 C1(NC(C2CCC(C)N2C(c2ncccc2Cl)=O)=O)CC2CCCCC12 Cn1nnc(C(=O)NCC2OCCC2C(N2CCC(CC3CC3)C2)=O)n1 c1(NC2CCCC(NC(c3ccc(C(F)F)cc3)=O)C2)ccc([N+](=O)[O-])c(O)n1 CCCCC(CN=c1[nH]c2cc(Br)ccc2o1)NC(=O)CCC1CCC(=O)NC1 C1(CC(=O)NCCc2cc(C)on2)(NC(C2CCC(C)(C)C2)=O)CCCCC1 N1(CCNC(c2ccc3cc[nH]c3c2)=O)CCCC2(C1)CC2(F)F N1(C(C2(C#C)CCN(C(c3cccnc3S)=O)C2)=O)CC(O)C2(CCCC2)C1 c1(SC)cccc(CC(=O)NC2CC2CNC(c2c(Br)n[nH]c2C)=O)c1 N1(C(=O)NCCN2CCOCC2)CCC(NCCc2ccns2)CC1 C1(NC(=O)OCCNC(C)=O)CC1C N1(C(C(CC)CC)=O)CCCC(C2CN(c3nnc(C(=O)OCC)s3)C2)C1 N1(C(C(=O)NCCCSCC)c2nc[nH]n2)CCC(Oc2ccccc2)C1 c1cc(C2CC2)ccn1.C1(COC)CC(C(=O)N)CO1.c1(C(=O)NC)cc(OC)n[nH]1 C=C(C)C(O)CC(=O)NCCC1CCN(C(C2(F)C3CCCCC23)=O)CC1 C1(CNC(C(c2ccccc2F)C)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)C1 C1(N(C(C(C)OCC#C)=O)C)CCCCC1NC(c1cc(C(C)C)oc1C)=O CCC(C)(CNC(C1CN(C(c2ccc(Cl)o2)=O)CCN1C)=O)C(N)=O c1(C(=O)NC2(COC)CN(C(C3CCCCCCC3)=O)C2)cnccc1C#N Cc1cc(CNC(=O)CCC2CC2)oc1C(=O)Nc1cnn(CC2CCC2)c1 N1(C(c2nc(C)c(Br)s2)C(=O)NCCSC)CC2CCC(C1)C2(F)F c1(NC(C2(C)CNC(=O)C2)=O)ccc2nccn2c1 CCC(CC(=O)N(CCNC(C1CN(C(C)C)C1)=O)C1CC1)OC N1(C(C2(OC)CC=CC2)=O)CC(c2ccccc2)CC1C(=O)O CC(C(CO)NC(=O)CNS(N)(=O)=O)NC(=O)CCN1CCOCC1 C1(NC(CCN(CC(F)(F)F)C)=O)C2CC1N(C(C1CCCCO1)=O)C2 C1(S(C)(=O)=O)(C(=O)NC(CNC(C(n2cnc(C#N)n2)CC)=O)C)CCCCC1 N1(C(CSSC)=O)CCC(CNC(c2c[nH]nc2OCC(F)F)=O)C1(C)C C1(C)(C(=O)NCC2C3CN(C(c4nc(CCC)sc4)=O)CC32)CCC(F)(F)CC1 c1(CN2CC(C(=O)NCCn3cccc3)C(O)CC2)c(O)ccc(F)c1Br c1(C(=O)NC(C(=O)NCc2nccs2)C2CCOC2)cnc(C2CC2)o1 c1(N(C(C)=O)C)ccccc1C(=O)NCC1CN(C(=O)CN(S(C)(=O)=O)C)C1 c1(CC(=O)NCC2CCC(CNC(C34CCC(CC3)C4)=O)CC2)ncccc1Cl C12(C(N(C3C(OC)COC3)C)=O)CCC(CN(C(=O)C(F)C(C)(F)F)C1)C2 c1(SC)ccc(N)cc1C(N1CCN(C(c2ccc(C)cc2C)=O)C(C)C1)=O C#Cc1cc(-n2cc(CC(=O)OC(=C)F)nn2)cc(F)c1 C(N=c1cc(NCc2cccnc2C(F)(F)F)nc[nH]1)C1(COC)CCCC1 C1(NC(CNC(C2CCC(CO)CC2)=O)=O)CN(C(C2CS(=O)(=O)C2)=O)C2CC12 C(=O)(C(C(C)NC(=O)CCC1CCC(C)O1)SCC)N1CC(CCC#C)C1 C1(NC(C2CCOC2)=O)C2CN(C(=O)C(c3cscn3)C3CC3)CC12 c1(CCC)cc(C(=O)NC2COCC2NC(C2(OCC)CCOC2)=O)cc(O)n1 N1(C(=O)OC(C)(C)C)CCCC(O)(C(=O)NC2CC(n3cccn3)C2)CC1 C(CC(C(=O)NC1(C=C)CC1)OC)NC(C1(COC)CC(=C)C1)=O n1(CC(=O)NCC2N(C(CC3N(C(C)C)CCC3)=O)CC2)ncc2cccnc12 O=C1CCC(CC(=O)NCC(O)CCNC(=O)Cc2csc(C3CC3)n2)C1 N1(C(CCc2c(C)noc2Cl)=O)C2CCC1CC(NC(=O)C(F)CC1CC1)C2 c1(NC(C2CCC(NC(CC(C=C)(C)O)=O)CC2)=O)c(C)ccn(C)c1=O c1(C(=O)NC2C=CC(CNC(C=CCOC)=O)C2)ccc(F)c(C2(C)CC2)c1 C(=O)(CCCCCCBr)N1CC(NC(c2cccc(C)c2I)=O)C(C#N)C1 C1(NC(c2ccc(Cl)c(F)c2)CO)CCC2CNCC12 c1(OC)ccc(C(N2CC(CNC(c3n[nH]c(C)c3O)=O)CC2C)=O)nc1Cl N1(C(=O)CC2OCCCO2)CCC(CO)(NC(=O)COCC2CCCC2)C1 c1(NC)cnc(NCC)nc1.CCC1CNC(=O)C2CC2C(=O)N1 C1(=CC(=O)NCc2cc[nH]c2C(=O)NCC2C3COCC23)CN2CCC1CC2 N1(C(C2(CC#C)CC2)=O)C2CCC1(CNC(=O)CCc1ccc(O)nc1)CC2 C1(F)(CNC(Cn2c(C)ncc2)=O)CCCN(C(=O)CCC(=O)c2ccc[nH]2)CC1 Cc1ccc(O)cc1-c1cccc(C2(C(=O)Nc3ccc(CO)nc3)CC2)c1 Cc1n[nH]cc1C=CC(=O)NC(C1CCN(C(=O)C(C)NC(=O)C2CC2)C1)(C)C c1(OC)ccc2c(c1)OCCC2NC(c1ccc2sc(=O)n(C)c2c1)=O CC1CC(C(=O)NC23CC(C2)N(C(C2(F)CCOCC2)=O)C3)c2ccccc2N1 C1(N(C(=O)CSCC(F)F)CC)CCCN(C(C2C(C)(C)C2(C)C)=O)C1 c1(C(=O)NCC(=O)NC(C(C)NC(CCOC(C)=O)=O)C)ccc([N+](=O)[O-])cc1 Cc1ccccc1C(C)C(N1CCOC(CNC(=O)CC2CC2C)C1)=O N1(C(c2c(Cl)cn(C)n2)=O)CC2CCOC2(CNC(=O)C(O)Cc2cnc[nH]2)C1 c1(C(N)=O)ccc(C(N2CCC2CNC(=O)CN2CC3CC3C2)=O)cn1 N1(C(c2c(C)n(C3CC3)cc2)=O)C2CCC1CN(C(c1ccnc(F)c1)=O)CC2 c1(C(=O)NC2CCC(CC(=O)NCC=C=C)CC2)c(C)nn(C)c1OC N12CCC(CC1)C2=O.C12(OCC)CCCC1C2.C1(COCCNC(=O)CO)CCCC1 c1(C(N2CC(CC)C2)C(=O)NCc2cnn(C)c2Br)cc(C(F)(F)F)ccc1F C(=O)(C1=NOC2(CCC2)C1)N1C(CC(=O)NCCCF)CC2(CC2)C1 C1(C(=O)NC2(C)CCN(C(=O)CCc3ncccn3)C2)C(O)C2CCOC12 C(=O)(CC(CC)N(C(=O)C(F)C(C)C)C)N(CC#CC)C.n1(CCC2CC2)cncn1 C1(CC)CN(C(c2cnn(C)c2)=O)CCN1Cc1ncc(Br)cc1Br CN1CC(C(N2CCC(N(C(=O)Nc3cncs3)CC3CC3)CC2)=O)CC1=O c1(CNC(CC2CC(NC(C=COCC)=O)C2)=O)ccncc1SC.c1(C)cccs1 CC1CN(C(c2sc(N(C)C)nc2Cl)=O)CCC1CNC(=O)C(C)(C)C#N Nc1ccc(CNC2CCC(C(=O)Nc3nc(O)cs3)C2)cc1[N+](=O)[O-] c1(C(=O)NCCN(CC(C)O)C(C2CC3CC3C2)=O)ncc(Br)cc1N Cc1nnc(O)c(C(=O)NCC2C=CCN2C(c2cnc[nH]2)=O)c1C C1(C(N2C(CN(C(C(CC3CCCC3)OC)=O)C)CCC2)=O)COC(=O)N1C C(=O)(C1CSc2ccccc21)N(CCC)CCNC(c1cnc(C(F)F)nc1)=O c1(OC)ccc2[nH]c3c(c2c1)CCN(C(=O)C(=O)NC1CCCC1)C3 Cc1nc2ccc(C(=O)NC(C)CNC(=O)CCC(C)(C)[N+](=O)[O-])cc2n(C)c1=O C(=O)(C(CC(C)C)C(C)C)NCC1(CNC(c2c(Br)ccc(C)n2)=O)CC1 C1(C(=O)NCC2(CNC(C3(C)CCCCC3)=O)CCC2)CCn2nnnc2C1 N1(C(C(C=C)OC)=O)CC2(CCN2C(=O)C(N2CCSCC2)C)C1 C(=O)(C#CC1CCCO1)NC1(CNC(CCCc2n[nH]c(=N)s2)=O)CCOC1 C12(NC(C(=O)NCCCNC(c3c(CC)noc3)=O)=O)CCC(CC1OC)C2 NS(=O)(=O)c1ccnc(C(=O)NCCCNC(c2conc2C2CCC2)=O)c1 c1(C(=O)NC2CCN(C(c3cncc(N)c3)=O)C3C2C3)cc2c(nc1O)CCC2 N1(C(c2occ(C)c2)=O)CC(C)CN(C(c2ccc(C#N)cc2O)=O)CC1C N1(C(CCOCC)=O)CC(CN(C)C(C2(C)CCC(F)(F)C2)=O)C2(CC2)C1 C(=O)(C(C)S(N)(=O)=O)NCC(C(C)C)(C)NC(C1CCCN2CCCC12)=O N1(CC)OCC(NC(C2CC(O)CN2C(=O)CCOCC(C)(C)C)=O)C1=O CCC(O)C(C)C(=O)NCC(c1cccc(Cl)c1Cl)NC(c1c[nH]c(=N)s1)=O C1(N(C(c2ncc(C)c(C)c2)=O)C)CCN(C(=O)C(O)CF)CC12CC2 C(CC(C)(C)C(=O)NC1CCCC(CNC(c2cnc(C(F)F)s2)=O)C1)OC c1(C(=O)NCC2(F)CN(C(CC(C(F)(F)F)OC)=O)C2)ncc2c(F)cccn12 c1(CC)cc(C(=O)N(C)CC2CCCN2C(c2cscc2SC)=O)c(C)o1 C(CCCC(C)C)(C(=O)O)N(C)C(=O)Nc1ccccc1OCC1CCCCO1 c1(OC)ncccc1CN1CCOC(C(=O)NCCc2cnc[nH]2)C1 c1(C(=O)Nc2ccc(Nc3nccc(C(=O)OCC)n3)cn2)ccnc(Cl)c1F C1(C(N2CCC(C(=O)NCCC3CC3CCCO)(CC)C2)=O)CC(=O)NC(=O)C1 C=C(Cl)CC(C(=O)NCC(C)F)NC(c1ccc(Cl)cn1)=O C(=O)(N=c1cc[nH]c2cc[nH]c12)C1C(NCc2ccc(C)s2)C1 N1(C(COC)=O)CCC2CCN(C(c3ccc(NC4CCSC4)cc3)=O)CC2C1 C(=O)(C(C)CC(F)(F)F)NC1(C(=O)NCC#C)CC(F)(F)C1 C1(CNC(C(C2CCCC2)OC)=O)CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 Cn1nccc1C(O)C(=O)NC(=O)C1CC1.C12CC(C1)C(=O)N(C1CCC1)CC2 C1(C(=O)NC(c2nc[nH]n2)CC)(CNC(=O)C=CCO)CCCO1 O=NN1CCCCC1C(N1CCOCC1CC(=O)NC1CCCOC1)=O C=C(C)C1OCCC1C(=O)NCC1(CNC(c2ccc(O)nc2)=O)CC12CCC2 c1(CC(=O)NC2CC3CC2N(C(C2CC4CC4C2)=O)C3)cnn2ccccc12 CC1CN(C(=O)CC2CCC3CC23)CCN(C(=O)CSCc2ccncc2)C1 N1(C(c2cccc(Cl)c2O)=O)CC2CCN(C(c3ncoc3C3CC3)=O)C2C1 c1(C(N2CCCC(C)C2CNC(C2CCN(C)C2)=O)=O)cc2n(n1)CCCC2 C(=O)(CC1=CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1)NC(c1c(C)ncs1)C N1(CC(N2CCC(NC(C(C)OCCOC)=O)C2)=O)OC(C)(C)CC1=O c1(C(=O)NC2CCN(C(c3cn(C(C)(C)C)nc3)=O)C2)cc2ccoc2cc1F C1(CCC(C)C)CCC(C(=O)NCCCNC(C2CCCC(N(C)C)C2)=O)CC1 Cc1ccc(=O)n(CC(=O)NC2CN(C(=O)C(c3cncnc3)C)CC2(C)C)n1 Cc1nc(CC(=O)NC23CC(C(=O)Nc4[nH]cnc4C(F)(F)F)(C2)C3)co1 N1(C(c2c(C)cc[nH]2)=O)CCN(C(c2cn(C)cc2C)=O)C2CCCC12 Cc1c(Cl)ccc(C(=O)N(CCCCCCNC(=O)COCCF)C)c1Cl C1(NC(CCc2cc(C(=O)OC)on2)=O)CCN(C(c2nocc2C)=O)CC1O C(=O)(C(F)CC(N)C(=O)OC)NCC(CNC(=O)C(F)(F)C(C)(C)O)OC N1(C(c2n(C)ncc2)=O)CC(NC(=O)CC2CCC(C(F)(F)F)CC2)C(O)C1 C12(OC)CCN(C1)C2=O.N1(CC(=O)NCC2CC(OC)C2)CC2CC2C1 Cn1cnc(CNC(=O)CCOCCNC(=O)CN=[N+]=[N-])c1 c1(NC(C23C(CN(C(C(C=C)(C)CC)=O)C2)C3)=O)cncc([N+](=O)[O-])c1 N1(C(c2ccc(CCC)s2)=O)CC(OC)C(NC(c2cscc2C(F)F)=O)C1 CC1CCCn2cc(C(N3CC(F)CC3CNC(=O)C=Cc3cc[nH]c3)=O)nc21 Cc1c(C(=O)N(CCCN(C)C(c2cc(C(C)(C)C)on2)=O)C)cnn1C1CC1 N1(C(C(C)C(C)O)=O)CCN(C(=O)CC2OCCC2(C)C)C2(CCC2)C1 C1(C2CCN(C(=O)C(c3cnccn3)C)C2)(NC(C2CCC(C)C2)=O)CC1 CCC(C(=O)NC1CCCCC1C(=O)NC1CC2(CCCCO2)C1)C(C)(C)CC Cc1cc(N2CCC(O)(C(C)NC(c3cnoc3)=O)C2)nc(C(C)C)n1 CC(CC(F)F)C(=O)N(CCC(=O)N(C)Cc1nc[nH]n1)C1CC1 c1(C(=O)NCC2N(C(C(C3CCOCC3)OC)=O)CCOC2)nnc(O)cc1O c1(C(CNC(=O)NC2CCSC2)O)c(F)cccc1F C1(C(=O)NC(C(C)SC)C)CCC(C)(C)N(C(=O)C(C)(C)CO)C1 c1(CCC(N2CCC(NC(COCCC=C)=O)C2C)=O)c(C)nc(O)nc1O N1(CC(C)NC(=O)C=CCN2CCCC2)CCN(C(=O)CCCF)CC1 C1(NC(CCC2N(C)CCCC2)=O)CCSC12CN(C(C1CC1(F)F)=O)C2 C1(C(C)C)CN(C(=O)CNC(=O)CC#N)CCCN1C(C1(c2ccncc2)CC1)=O C1(C2(O)CCC2)(C(=O)NC(C=CC(=O)N(CC)Cc2cccnc2)(C)C)CC1 c1(C(CC)C)ccc(C(N2CCC(NC(=O)CC3(C)CC3(F)Cl)C2C)=O)cc1 C1(CNC(C2CN(C3(C)COCCO3)C2)=O)CC2(CC(NC(=O)C3CC3)C2)C1 C1(NC(C2CC3(C2)CC3F)=O)CC2COCC(C1)N2C(C1CC2(CCC2)C1)=O C1(F)(CNC(CN(C2CCSC2)CC)=O)CC(CNC(=O)CN(C)C2CC2)C1 C1(C(=O)OCC)CCC(C(=O)NCC2(CC(C)C)CCC2)C1 N#Cc1nc(NC(C2(C(=O)N=c3cc[nH][nH]3)CC2)=O)ccc1Cl c1(C(=O)NCC2N(C(C(CC)F)=O)CCN(C)C2)ccncc1[N+](=O)[O-] c1(N(C(CN(CC(C)O)CC(N)=O)=O)CCCCCO)cccs1 c1(CC(=O)NCC(C)(C)CC2CN(C(C3CC3C3CCC3)=O)C2)ccc(F)cn1 c1(C(N2CCC(O)(CNCc3c(OCC)cccn3)C2)=O)cc([N+](=O)[O-])n[nH]1 N1(C(C2(N(C)C)CCCSC2)=O)CCC(O)C(NC(C2CCC2)=O)C1 CCC(C(=O)N1CCC(N(C(=O)CC2CC(C)(C)C2)CC2CC2)C1)n1ccnc1 N1(C(C2(OC)CCC2)=O)CC(NC(c2c[nH]c(=N)s2)=O)C(CC2CC2)C1 Cc1ccc2oc(N3CCCC4(CC3)CC4)nc2c1 C1(CNC(CC=CC)CO)CC(F)(F)CN1C(c1ccnc(F)c1)=O c1(NC(c2n(CCCCCC)nnn2)(CSC)CC)cccnc1C N#Cc1cncc(CN2C(C(=O)NCCCF)CC3CC23)c1 c1(CC(=O)NCC(CCNC(c2ccn(C)n2)=O)O)ccccc1S(C)(=O)=O C1(CNC(c2cc(C3CC3)[nH]n2)=O)CC2COCC2N1c1ccccc1[N+](=O)[O-] C(=O)(C1=CCN(C(=O)CSC(F)F)C1)N1CCC(=CCC)C1 C1(CNC(N(C(C)C(=O)NO)C2CC2)=O)CCCC(C)(C)C1 c1(C(N2CCCC(CC(N)=O)C2)C(=O)NC(CC)C)cc(C)nn1CC Cc1cc(CC(=O)NC23CC2CN(C(c2ccc(CO)o2)=O)C3)cc(F)c1 N1(C(CNC(C(C)NC=O)=O)=O)CCC(C)(C)C1C(=O)NCCO N1(C2C(NC(CC(=O)NC3CC3)=O)CCC2)CCN(C(=O)CCC2CCC2)CC1 C(=O)(C#CC1CCC1)NC1C(CCC)CN(C(=O)C(CC2CC2)OC)C1 N1(C(CCCC=C)=O)CCC2CC2(NC(C2CCN(OC)CC2)=O)CC1 C1(CNC(C(c2c(C)ccnc2)(C)C)=O)CCN(C(=O)C(C)CN(C)C)C(C)C1 N1(C(C2CC(=C)C2)=O)CCC(N=[N+]=[N-])(C(N2CCC(c3nn[nH]n3)C2)=O)C1 c1(C(N(CCNC(=O)Cc2ccccc2)C2CC2)=O)ccc(C2CC2)nc1 C(CCC(C)C)NC1C(C(=O)NCCCNC(CCN(C(C)=O)C)=O)C1 C(=O)(CCCCCF)N(C1CCCC1)CCNC(C1CS(=O)(=O)C1)=O S(=O)(=O)(CCS(=O)(=O)NC(=O)NCc1ccc(Br)c(F)c1)Nc1ccccc1 CC1CCC(CC(=O)NCC(C)N(C(=O)CC(C)n2cccc2)C)C1 C1(NC(CC)=O)CCCCC1NC(=O)Cc1cc[nH]c1 N1(C(C(CC)n2ccnc2)=O)CCC2C(C(N3CC(N(C)C)C(C)(C)C3)=O)C2C1 C1(C(=O)NC(C)CNC(c2ccc(Cn3ccnn3)cc2)=O)CC2CC1CC2O C(=O)(C(CNC(=O)CC1CC1)N(C)C)NC(c1nccn1CC)CC N1(C(CC(C=C)(C)C)=O)CC(C)N(C(C2CC(C(=O)OC)C2)=O)CC1C N1(C(C2CN(CC)C(=O)CC2)=O)CCC(C(F)F)C12CC2 C=CCC(C)(CNC(C1CCC(C)N1C(c1cn(C2CC2)cn1)=O)=O)CO c1(C(=O)NC2(C)CCCN(c3ccc(NC(N)=O)cn3)C2)ccc(F)c(C#N)c1 Cn1c(O)nc2cc(C(=O)NC3CCC(NC(C4CC4C#N)=O)C3)ccc12 Cc1cc(C(=O)NC2CCCCCC2C(=O)NCc2ccsc2C)cc(O)n1 c1(C(N2C(C)CC(CNC(c3nc(COCC)sc3)=O)C2)=O)cnc(O)c(C)c1 C(=O)(C(CC(F)F)OC(F)F)N1CCC(CC(C)NC(=O)COC(F)F)CC1 c1(C(N(CCN(C(CCOCC)=O)C(C)C)C)=O)c(N)cc(F)cc1Cl N1(C(C(CC)n2ccnc2)=O)CCC(CN(C(=O)CC(C)C2CCCC2)C)CC1 CC1CC(C)(C(=O)NCC2(CNC(=O)Cn3ncnn3)CC2)c2ccccc2N1 C1(NC(C2CCN(C)C2=O)=O)CN(C(c2cc(C#N)c[nH]2)=O)CC2(CCC2)C1 N1(C(C2(CNC(C3CC4CC4C3)=O)CCCO2)=O)CCC2(CCCO2)C1 N1(C(C(C)CNC(C2CCCC23CCC3)=O)=O)CCC2(CC1)CC2C#N C=CCCC(C)(C)C(=O)NC(C)CN(C)C(C12CC(c3ccccc3)(C1)C2F)=O N1(C(C#CC2(CC)COC2)=O)CCC2(CC1)CCN(C(=O)CN1CCC1C)C2 N1(C(CN(C)C2CC2)=O)CCCC(CNC(C2C3C(=O)OCC23Br)=O)CC1 c1(C(N2C(C(CNC(CCCC)=O)(C)C)CCCC2)=O)cc(C#N)c(N)cc1O c1(C(N2CCC(CCN3CC(=O)NCC3)C2)=O)cn2cccc(Cl)c2n1 c1(C(C)C)ccc2occ(C(N3CC4CN(C(=O)C5=COCC5)CC4C3)=O)c2c1 CCCC(C(=O)NCCN(C1CCCC1)C(c1nnc2ccccn12)=O)C(C)C C1(C)(NC(C(CC=C)NC(=O)C=C(C)c2ccco2)=O)CC2CCC1C2 N1(C(c2c(OC)ccs2)=O)C2CCC1CC(CNC(c1ccccn1)=O)C2 C1(COC(=O)NCc2cccc(Cl)c2)CC2(CCN(C(=O)C3CC3)C2)CO1 C(=O)(CCC(C)S(C)(=O)=O)NC(CCCC)CNC(=O)C(C)CCN(C)C C=Cc1cncc(C(N2CC(C(O)C(=O)NC3CN4CCCC3C4)C2)=O)c1 Cc1cnc(CNC(C2C=CCN2C(=O)CC(C)N(C)C)=O)c(C)c1 C(=O)(CS(=O)C(F)(F)F)N(CCCNC(=O)CCc1cncn1C)C N1(C(c2c(C)scn2)C(=O)NC(C)C)CCn2ccnc2C1C CCCCC(C(=O)N1CC2C(CNC(c3coc(O)n3)=O)C2C1)N(C)C N1(c2ncc(C)nc2)CCC(C2CCCNC2)CC1 C(=O)(C(O)CC(F)F)NCC(CC)NC(c1scc(OC)c1OC)=O N1(C(c2ccccc2)=O)CC2C3CCC(C2C1)N(Cc1cc(C2CC2)on1)C3 NS(=O)(=O)C1CCCN(C(=O)C(=O)NC2CCCCC2C(F)(F)F)CC1 C(=O)(C1=CCC(C)CC1)OC.C(=O)(CC(C)C(=O)OC)N1C2(C=CC1)C(=O)NC2 C1(O)(CNC(C2CC(C)(COC)C2)=O)CCN(C(=O)COc2ccccc2C)C1 c1cc(Cl)nc(C)n1.C(C)(C=O)OCCCC.C1(=O)NCCN(CC)CCN1 N1(C(C2C3CCC(F)(F)C23)=O)CC2(C1)CN(C(C1(C3CCCO3)CCC1)=O)C2 Cc1cccc(C(=O)N(C(CNC(C2(C)CCCCO2)=O)C2CC2)C)c1 N1(C(Cc2ncc(C)o2)=O)CCCC2(NC(=O)Cc3ccc(F)cc3)CCCC12 CC1SCCCC1C(=O)NCc1cc(C(=O)N(C2CCOC2)CCF)n[nH]1 Cc1cccc(CC(=O)NC23CC(C(N4CCC(O)(CO)C4)=O)(C2)C3)n1 C(=O)(C1OCCc2ccccc21)NCC(CO)NC(c1ncn(C)n1)=O C(=O)(C#CC1CCCCC1)NC1C(CC)CN(C(c2coc(C(F)F)n2)=O)CC1 N(C1CCCc2c(F)cccc21)C(C(=O)NC1CCCN(CC(F)(F)F)C1)=O C=CC(C)(CCOC)C(=O)NCC(CC)N(C)C(c1ccns1)=O CCC(C(=O)NCC(N1CCN(C(C2CCOCC2)=O)CC1)=O)C(C)C c1(C(N2CCC(N(C(=O)C(C)(O)CC)CCCC)CC2)=O)ccc2oncc2c1 C1(C(C)C(=O)NCCCC2CCCC2)CCN(C(C2CCCC2)=O)CC1 C(=O)(C(O)CCCNC(=O)C1=NNC(=O)C1)NCC(C)OC C(C1C(=O)CCNCC1C)NC.COC(C)C c1(CNC(C2(C)CC(=C)C2)=O)cccc(CNC(=O)CC2CCCN(C)C2)c1 CC(C)CC(C(=O)NCCOC1CN(C(=O)C(C)C(C)O)C1)N1CCCCC1=O N1(C(CC=CC(C)(C)C)=O)CC2C3CCC(C2C1)N(C(=O)C(F)C1CC1)C3 c1(N(C(C2CC(OC(C)=O)C2)=O)C(C2NCCC2(C)C)=O)ncccc1F c1(N2CC(CC(C)NC(=O)CCc3ccc(Cl)cc3)C2)ccc([N+](=O)[O-])c(O)n1 C1(NC(c2csc3nccn23)=O)CS(=O)(=O)C2CN(C(=O)CC3C=CCC3)CC12 C(=O)(C1=C(Cl)CCCC1)N1C(C(=O)NC(CCCCC)C)(COC)C=CC1 c1(C(N(CCNC(CCNC(=O)OC)=O)CC2CC2)=O)ccc(C(F)(F)F)nc1C N1(C(C(CC=C)NC(C)=O)=O)CC2(CC(NC(c3c[nH]nc3OC)=O)C2)C1 C1(CC(=O)NC(CCSC)C)CN(C(c2ccncc2N)=O)CCO1 c1(C(N2C(CNC(c3ccc(CC)s3)=O)CC3CC32)=O)cccc(O)c1Cl Cc1[nH]nc(C(N2CCC(NC(=O)Cc3cccnc3O)C2C(C)C)=O)c1Cl N1(C(C)=O)CCN(C(c2cc(-c3cn(CC(F)(F)CO)nn3)co2)=O)CC1C S(=O)(=O)(c1ccc(NC(C)C2CC2)cc1Cl)NC(n1cccn1)C C1(C(N(C2CCCCC2C(C)(C)C)C)=O)CCCN(Cc2ccccc2)C1 N1(C(c2cn(CCC)nc2)=O)CCN(C(=O)Cc2ccc(C)s2)C2CCCCC12 CCCCS(=O)(=O)NC(C)C(=O)NC1CCN(C(=O)C=Cc2cccn2C)C1C CCS(=O)CC(=O)NC(CCN(C)C)C(=O)NCC(N1CC=CC1)=O c1(C(N2C(CNC(c3c(C)nc[nH]3)=O)COCC2)=O)ccc2ccncc2c1 C1(NC(c2c(NCC)cccn2)=O)CN(C(C2CCC3CC3CC2)=O)CCC1F c1(C(=O)NCC(CC)NC(c2cc(C(C)C)ccc2F)=O)cnc(O)c(C)c1 c1(C(=O)NCC(CC)NC(c2scnc2C(C)C)=O)cc(F)cc2c1CCC2 CCCC(C)(O)C(=O)N(CCCCCNC(c1[nH]c(C)nc1CC)=O)C c1(SCC)ccc(NC(C2(NC(c3cn(CCO)nn3)=O)CCCC2C)=O)cn1 C1(C(N(C2CC2)CC2N(C(C(C)OCC=C)=O)CCC2)=O)CCC(CO)CC1 CCC(C)CC(C)N=c1nc2scnc2c(NCCCn2nccc2C2CC2)[nH]1 c1(CNC(CCC2CCC(NC(C(C)OC(C)(C)C)=O)C2)=O)cnn(C)c1O N1(C(c2n(COC)ncc2)=O)CCC=C(C(=O)Nc2cnc(Cl)nc2C)C1 C1(CC=C)(NC(=O)CCOC)CCN(C(=O)C=Cc2csc(Br)c2)C1 C(=O)(CCCC(=O)NCC1(C(N2CCC2(C)C(=O)OC)=O)CCCCC1)NCC C(CC1c2ccccc2CCN1C(C1CCSC1)=O)NC(C(CCC)(C)CC)=O CS(=O)(=O)c1cc(C(=O)NC23CCC(CC2)N(C(=O)Cc2cscn2)C3)co1 c1(CC)nn(C)c(CC)c1C(N1CC(NC(C2CC=CCO2)=O)C(C)C1)=O N1(C(CCCC=C)=O)CCC2CN(C(=O)C#CC3CCOCC3)CCC2C1 CN1CCC(CN(C2(CO)CC(F)(F)C2)C=O)C1c1ccc(Cl)cc1 c1(SC)nc(Cl)cc(=NCC2CCCC(NC(=O)CSc3nncn3C)C2)[nH]1 C1(CC)CCCN(C(C2C3CCCOC23)=O)C1C(=O)NC1CCNC(=O)C1 n1(CC(N2CC(NC(c3scc(C(C)=O)c3)=O)C(OC)C2)=O)nc(C)c(Cl)c1C C12CC(C13CCC3)C(=O)N2.C1(C(=O)OC)CC2CCCCC12 Cc1ccc(C=CC(N2CC3CC(CNC(C4(F)CCC4)=O)C3C2)=O)cc1Cl C(C)(CCCN=c1ccc(S(=O)(=O)N2CCCC2)c[nH]1)NC(C(CSC)(C)C)=O C(=O)(C(C)C1=CCCC1)NC(CC=C)CNC(c1cnsc1C)=O c1(SCC(C)O)ccccc1N1C(=O)COc2cc(Cl)c(F)cc21 c1(C(=O)NCC2CCCN(C(C(COCC)C)=O)CC2)cccc2[nH]ncc12 c1(C(C)CNC(=O)C(=O)NC(Cn2cccn2)C(=O)O)ccc(C(F)(F)F)cc1 N1(C(c2ccn(CC)n2)=O)CC2CCC2(C(=O)N(c2cccc(C)c2)C)C1 N1(C(C(C)CC(N)=O)=O)CCCC2(CCCN2C(=O)Cn2cccc(C)c2=O)C1 CC1(Nc2ccc(O)nc2)CCC(C(=O)O)CC1 c1(OCC)cccc(C(N2CC(NC(C3(C(F)F)CCCOC3)=O)C(C)C2)=O)c1 C1(C2CN(C(c3nnccc3C)=O)C2)(NC(C2C(CCC)C2)=O)CC1 C(=O)(CC(C)(O)COC)NCC(c1cccc(F)c1)NC(COC)=O N1(C(CC2(C)CC2)=O)CCCC(NC(C2CN(C(C)C)CCO2)=O)C1 Nc1cc(C(=O)NCC2COCC2NC(=O)C=Cc2cccs2)c(F)cc1F c1(C(=O)NC(CNC(CCOCC#C)=O)(C)C(C)C)ccc2c(c1)CCC(C)N2 c1(C(=O)NC2CN(C(C3CN(OC)C(=O)C3)=O)CC2C)cc(F)c2[nH]nnc2c1 CC(C1=CCN(C)CC1)NC(C1(NC(=O)OC(C)(C)C)CC1C)=O C12CCN(C1)C(=O)C(=O)COCC(=O)N2.C1(C#N)(C)CCC1.CO c1(C(=O)NC(c2ccccc2)C(C)C)ccc(CNC(C2CCC(NC)C2)=O)nc1 Cc1c([N+](=O)[O-])cccc1S(=O)(=O)NC1CS(=O)(=O)C2CNCC12 c1(SC)ncc(Br)c(N2CC3(CN(C(=O)CC4CCC5CC45)C3)C2)n1 C=C(CNC(C1(C(C)C)CCN(C(c2cnn(CCO)c2)=O)C1)=O)C(F)(F)F c1(C(=O)NCCCCNC(=O)Cc2cccc(F)c2F)noc2cc(Cl)ccc12 c1(CNC(C(c2nnn(C)n2)N(CCN2CCCS2(=O)=O)CC)=O)cccc(Cl)c1 c1(CNC(c2n(CC=C)nnn2)c2ccnn2C2CC2)ccc(F)cc1Br c1(OC(C)C(=O)NC2CC(CNC(C3(O)CCSC3)=O)C2)ccccc1 N#CC1(C(N2CCC(C3CC3)(NC(c3cccc(Cl)c3)=O)C2)=O)CC2CC2C1 N1(C(C(C(C)C)O)=O)CC(NC(c2cccn(C)c2=O)=O)C(C2CC2)C1 c1(C(=O)OC(c2ccccc2)(CC)C)c(-c2ccccc2F)noc1C N1(C(C(C2CCC2)OC)=O)CCCN(C(C2CN3CCCN2CC3)=O)CC1C c1(C(=O)NC(C(C(=O)NCCn2c(C)cc(C)n2)C)C)ccc(C#N)cc1 N1(C(C(C)CC2CC2)=O)CC2CC(C(=O)NCC3CC(CC4CC4)CO3)(C2)C1 C1(C2CC2)(NC(c2cnnc(O)c2)=O)CCN(C(c2cc(Cl)c(F)cc2F)=O)C1 C#CCCCCCCCC(=O)NC1CCC(NC(C2(C3CC3)CC2)=O)C1 C(=O)(C(C(=O)N1CCC(N(C(c2ccc[nH]2)=O)CC)CC1)C(C)(C)C)OCC CC1(CNC(C2(F)CCN(C(c3cc(CO)on3)=O)C2)=O)CCOCC1 Cc1oc(S(C)(=O)=O)cc1C(N1CC2CC2(NC(=O)CC(C)(O)C2CC2)C1)=O O(NC(=O)C(CCN(C)C)N(C)C=O)C(C(=O)NC(C(C)C)CO)CC(C)C N1(C(C(C(C)C)NC(C2(C#N)CC(C)C2)=O)=O)CC2(C1)CC(C)(O)C2 c1(C(N(CCCN(C(CC2CCC(C)C2)=O)C)C)=O)ccc(S(N)(=O)=O)cn1 CCC(CC(=O)N1CCN(Cc2ccc(CC(=O)NC3CC3)cc2)CC1)C(F)F c1(C(N2CC3C(CNC(C(CC#C)C)=O)C3C2)=O)cccc(Cl)c1F N1(C(c2ncc(C(C)(C)C)s2)=O)CC2(NC(=O)Cc3ccncc3)CC1C2 CN(C)NC(=O)CCC(=O)NCc1ccsc1C(N1CCC(F)(CO)C1)=O CC1(C)CC(C(N2CC3CC3C3CC23)=O)CN1C(c1ccnc(CO)c1)=O c1(C(=O)OC)cc(CC(=O)NCCN(CC(C)O)C(C2CC2(Cl)Cl)=O)cs1 C(=O)(CCCCCNC(C1CCCC1CC)=O)NCC(CC)CCO c1(C(CNC(CC2(N)COC2)=O)(F)F)ccccc1 N1(C(C(F)=C(C)C)=O)CC(CNC(=O)C=CI)N2CCC1C2 C1(CN(C)C(C2(C(F)F)CC2)=O)C2CN(C(C3(F)CC=CC3)=O)CC12 Cc1cc(C(=O)NC2CCN(C(c3csc(C(F)F)n3)=O)CC2CO)c(C)cn1 C12NC(=S)N(C)C(CC)=C1C(=O)CCc1ccc(c(OCCOC)c1OCO)N2 Cc1cc(Br)c(C(N2CCCC(CNC(=O)COC3CCCC3)C2)=O)cc1F C1(CC(=O)NCCN(C(=O)C=C2CCOCC2)C)CCS(=O)(=O)C1 c1(C(=O)NC(C)(C)CNC(=O)C(O)C(C)(C)C)ccc2sccc2c1 C(N=c1cc(C)nc(N(C)Cc2nnc(C)s2)[nH]1)c1c(F)cc(C)cc1Cl C(=O)(CC(C)C(=O)OC)NC1(C(F)(F)F)CN(Cc2ccncc2C(F)(F)F)C1 CCC(C)C(C(=O)NCc1ocnc1C(N1CC2CCC1CC2)=O)N(C)C C(=O)(CN=c1cc[nH]cc1)NCC1(C)CC(NC(c2ccc(Cl)cc2)=O)C1 C1(C(=O)NC2CCN(C(Cc3nnc(C)s3)=O)C2C2CC2)CCn2nccc2C1 CCCCCCCCNS(=O)(=O)CC1CCC(C)CO1 N1(C(c2cc(COC)no2)=O)CCOC2CCN(C(C3(C)CCCC3)=O)CC12 N1(C(CNS(CC)(=O)=O)=O)CCOCC(NC(=O)C(c2ccc(F)cc2)(F)F)C1 N1(C(c2cc(CC)nnc2C)=O)CC2(CCCC2NC(=O)CCC2CC2(Cl)Cl)C1 C(=O)(C1=C(C)CC(C)(C)CC1)N1CC(N(C(c2ccc(C=C)cc2)=O)C)C(F)C1 c1(C(N2C(CC=C)(C(=O)NC3CCOCC3=C)CCC2)=O)cc(C)c(C)nn1 Cc1cc(CN2CC3C(C2)N3C(c2ccc(-c3ccccc3)nc2)=O)cc(F)c1 N1(C(C(CC2CN(C(C(C)CN(C)C)=O)C2)F)=O)CC(C)OCC(C)(C)C1 C(=O)(CCCC(C)NC(=O)C(C1CC1)SC)NC(c1nc(CC)[nH]n1)C C(C)(C)(CC(C)N=c1[nH]c(=NCc2nnc3ccccn23)[nH]c2c1COCC2)OC N1(C(c2nc(C)c(Br)cc2)=O)CC2(CCC(C(=O)Nc3c[nH]nc3C#N)O2)C1 C1(C(=O)NC2CC(C)N(C(C3CC4(C3)CC4F)=O)C2)CC2CCCC(C1)C2=O N1(C(=O)C=NO)CCN(C2CN(C(=O)COc3ccccc3F)C2)CC1 C1(CCOC)CN(C(=O)CCNc2ccccn2)CCN1C(=O)C1=COCCO1 C(=O)(C1COc2ccccc21)NC12CN(C(c3c(C(C)C)scn3)=O)C(CC1)C2 c1(C(=O)Nc2c(NC(c3cnc(NC(C)=O)o3)=O)c[nH]n2)nn(C)c2c1CCC2 Cc1cccc(C=CC(N2CC3(CC3)CC2C(=O)NCc2cccc(Cl)c2)=O)c1 c1(C(N2CCC(NCc3c(Cl)ccc(OCC)c3)CC2)=O)ccc(O)c(C#N)c1 C1(C)(CN(CC=C)CC2CCCO2)CCC(NC(c2ccc(C)c(F)c2)=O)CC1 C1(NC(C(COC)C)=O)CN(C(C23COCC2C3)=O)CC1CSC N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CC=CC(NC(=O)CC2CCCC2(F)F)C1 O=C(C1=CCCN(C(=O)CCc2ccncn2)C1)N1CCOCC1CCO C1(CC)CN(C(=O)CC2(C)CC2(F)Cl)CCC1CNC(c1c(C)nn(C)c1Cl)=O C(C)(C)(CCCC(=O)NC(C)C(C)C(=O)C(c1c(OC)ccs1)=O)NOC c1(C(=O)NC2C(C(=O)NC(CC)CO)CCC2)cc(F)cnc1O C(=O)(CC(C)C(C)(C)NC(=O)CN1CCSCC1)NC(CC)CCCO Cc1cccc(C)c1NC(N1CCC(C(C)CNC(c2nccs2)=O)CC1)=O C1(NC(=O)CCCC2CCCCC2)CCN(C(c2ccsn2)=O)CC1CO c1(C(N(CC(=O)N(C2CCOC2)C)CC)=O)ccncn1 N1(C(c2c(CC)nns2)=O)CCN(CCNC(=O)Cc2csc(C3CC3)n2)CC1 c1(C(=O)OCC(c2cccc(Cl)c2)F)cc(Br)c2ccccc2c1 c1(NC(C2C(C(=O)Nc3ccc(C(=O)NC)cc3)C2)=O)cc(OC)c(F)c(F)c1 Nc1ccc(O)c(C(=O)NCC2CCCN(C(=O)Cn3cc(Cl)cn3)C2)c1 c1(C(=O)NCC2(CSCC)CC2)ccc(NC(c2ncnn2C2CC2)=O)nn1 c1(-c2cn(CCCC(=O)N3CC(N4CCCC4)C3)nn2)cncc(O)c1Cl c1(C(C(=O)NCCN(C(CC(C)n2cccn2)=O)CC(C)O)=O)ccc(O)cc1 CC(C(C(=O)N(CCCF)C)NC(=O)OC(C)(C)C)c1ccccc1 c1(C(=O)NCCN(C(C2C(C=C)OCC2)=O)C2CC2)nccc(OC)c1OC C(C(=O)N(C)CC1(C(=O)OC)CC1)(C(C)C)SCC.C1(=O)C(C)N1 C(=O)(C(O)CN(C)C)NC(C1CCCN1C(=O)CNC)C.c1(NC(=O)N)ccco1 C1(=CC(=O)NCCCC(C)NC(CC=C)=O)CCC(C)CC1 C(=O)(CS(=O)(=O)Cc1ccccn1)NCC(COC(=O)NC(C)(C)C)(C)O C1(C(N(CCNC(c2n(CC)c(O)nc2)=O)C)=O)CCC(N=[N+]=[N-])CC1 C1(CNC(=O)Cc2nc(C)n[nH]2)CCCCN(C(c2cc(Cl)ccn2)=O)C1.c1ccco1 N1(C(=O)OC(C)(C)C)CC2(CCOCC2)CC1CNC(C1CCC(=O)N1)=O C(=O)(CC(C)(C)C)NC(C)C(=O)NC(C1CCCCC1)CNC(c1ccncn1)=O Cn1ncc2c(N3C4CCC3CN(C(C3(C(F)F)CCCC3)=O)C4)nc(Cl)nc12 Cc1cc(C(=O)N(C2CCN(C(=O)C(C)C(C)C)C2)CCO)cc(C)n1 C1(C(C(=O)NCCCC(C)O)NC(C2C(CC)(CC)C2)=O)CCOC(C)(C)C1 c1(NC)cccc(C(=O)NCCC2CC(NC(=O)C(C)NC(C3CCC3)=O)C2)c1 N1(C(c2nc(C(C)=O)sc2)=O)CCC2(CC1)CC2NC(c1cnn(C)n1)=O Cc1cc(C(=O)NC(C(C)NC(c2ccsc2C(F)(F)F)=O)C(C)C)c(O)nn1 N1(C(c2cc(C)nc(O)c2)=O)CCC12CCCN(C(C1CC1C)=O)C2 C1(CCNC(CC(=C=C)C)=O)CCN(C(c2nccc3[nH]ccc23)=O)CC1(F)F N1(C(C(=O)NCCC#N)CC2CCCO2)CCC(Cn2cccc2)CC1 c1(CC(=O)NC(CNC(C(c2c(C)cncc2)C)=O)C)cccc(O)c1F c1(CC)cccc2c(C(=O)NC(C)(C)CNC(C3(CC)CC3)=O)c[nH]c12 c1(N(C)C)cccc(C(=O)NC2CCCCC2NC(=O)C#CC2CC2)c1 c1(C(=O)NC(COC)CC(=O)NCCCN2CCC(O)C2)cc2cccnn2c1 C1(NC(CSCc2cn(C)nc2)=O)COCCN(C(C2CC2C#N)=O)C1 C1(C(=O)NC(C(C)SC)C)COCCC1NC(=O)C(C(C)C)N(C)C Cc1nc(O)[nH]c1C(=O)NCC(C1CCC1)NC(=O)C(F)Cc1ccccc1 Nc1sc2cccnc2c1C(=O)NCCCCNC(C1CCC=CCCC1)=O c1(C(=O)NCCC(C)NC(c2c(C)ccn2C)=O)cn2nc(C)cc2[nH]c1=O N1(C(CC2N(C)CCOC2)=O)CC2CCC(C1)N2C(=O)CCC1CC1(C)C N1(C(c2c(C)ncnc2)=O)CC(NC(=O)C=Cc2cn[nH]c2)CC12CCCOC2 c1(NC(NOC2(C)CC=CCC2)=S)ccc2oc(C(N)=O)nc2c1 C(C(CC(=O)N1CCC(C(C)(C)NC(c2cnc[nH]2)=O)CC1)C(F)F)N(C)C Cn1c(CO)nnc1C1CCCOC1CN1CCC(Oc2ccncc2)C1 Cc1cccc(Br)c1OCC(=O)NC(C)CCN(C(=O)C1=CCC1)C N1(C(COCCCOC)=O)CCCCC1C(=O)NCCc1ccnc(C)c1 N1(C(C2(CC)CCOCC2)=O)CCC2CN(C(=O)CCCC#N)CC2C1 CCCCC(O)CCC(=O)NCC=C1CCN(C(C2(C)CCCC2C)=O)CC1 N1(C(CN(CCC)C)=O)C2CCC1CC(O)(CNC(C1C3CC3C1)=O)C2 C(N=c1[nH]c(N2Cc3c[nH]nc3C2)nc2c1CCC2)c1c(C(C)(C)C)n[nH]c1 c1(C(=O)NC2C3(CCN(C(C4C(=C)C4)=O)CC3)C2)cc2ncc(C)cn2n1 C1(NC(c2nc(CC)sc2)=O)CN(C(=O)C(C)CC2CCC2)C(C)(C)C1 O=C1OCCN(Cc2cccn3nccc23)C12CCC2 N1(C(c2ccc(NC(C)=O)s2)=O)CCCC(F)(CNC(C2COC(C)C2)=O)C1 CC1(NC(c2nocc2Br)=O)CCN(C(C2COCCO2)=O)CC1 N1(C(c2c(CC)onc2)=O)CCC(N(C)C(c2cnc(Cl)[nH]2)=O)CC1 c1(C(=O)NCC2C(C)(C)CCC2)n[nH]c2c1CN(C(C1CC(N(C)C)C1)=O)C2 C1(C(=O)NC(C)C(C)(C)NC(c2nnn3ccccc23)=O)CCc2nn[nH]c2C1 C1(C(=O)NCc2c(C(=O)NCC(C)O)cccn2)CN2CCC1CC2 Cc1nc(C(=O)NC2CC3CN(C(C4(CO)CCC4)=O)CC3C2)ccc1[N+](=O)[O-] C1(C(C)C(=O)NC2(CC#N)CCC2)CCCCC1 C1(NC(CCCCC=C)=O)CC2(C1)CC1(CC(NC(C3(C#N)CCOC3)=O)C1)C2 C1(OC)CN(C(=O)C(C)O)CCC1NC(c1sc(Cl)c(Cl)c1C)=O C(=O)(CC(C)(C)C)N1C(CNC(C)C(=O)N2CC(NC(=O)C3=CSCS3)C2)CCC1 c1(C(N2CCN(CCNC(CC3C(C)CCO3)=O)CC2)=O)cnc2ccoc2c1 C1(N(C2CC3CNC2C3)C(c2nc(CC)oc2)=O)CCN(C)C1C N1(C(c2cc(CC)nn2C)=O)CCC(F)CC1C(=O)NCC1(C)CC2(CC2)C1 C(=O)(C(CC)C(C)(C)CC)NCCN(CCC)C(c1cc(C)n(C2CC2)n1)=O C(C(=O)N1CC2CC(C1)C2NC(=O)C(C)CC(C)C)(C(C)(C)C)OC N1(C(C(C2CCCC2)OCC)=O)CC(O)(CCNC(=O)C(CC)n2cncn2)C1 c1(OC)ccc(CN=C(NCC(F)F)NCC2(c3ccnn3C)CC2)cc1 c1(C(=O)NCC#CC(=O)NCCCN(C)C)cc2cnccc2[nH]1 C(=O)(CC(O)CNC(=O)Cc1cnoc1)NCC(C1CCC1)OC C(CC(F)F)(C(=O)NCc1cncn1CC)NC(c1c(C)nc(CC)o1)=O C1(NC(c2ccc(SCC)cc2)=O)CC(C)CN(C(=O)COCC2CCCO2)C1 N1(C(COCCNC(CC)=O)=O)CCN(CCC2CCCO2)CC1 C(=O)(CCCn1cc(C2CCCC2)nn1)N(CCCc1ccsc1)C C(CNC(=O)COCCOC)(CC)(CC)NC(C1(CC)CCCC1)=O c1(C(CC(=O)N(c2ccccc2F)CCC#C)O)cccc(F)c1 C1(C(=O)NCc2cccc(C(=O)NC3(CC)CCC3)n2)CC2(CCO1)CC2 Cc1c(C(=O)NC2CC(N(C)C(C3SC4C=CC3CC4)=O)C2)[nH]c2ccccc12 N1(C(CC2(CNC(C(C)Cn3ccnc3)=O)CC2)=O)CCCC(O)CC1 c1(C(=O)NC2(C)CN(C(=O)COC(F)F)C2)ccc(=O)n(-c2ccc(Cl)cc2)n1 N1(CC(=O)N(C(C)CNC(=O)Cc2cnc[nH]2)CC)CCCS1(=O)=O C1(CC=C)(C(=O)N(C)CCOC(C)=O)CCCN1C(=O)CCOCC O(C1CCOc2c(Br)cccc21)C(C1CC(CC2CC2)C1)=O N1(C(c2occ(C(N)=O)c2)=O)CC(NC(C2C3CCCC23)=O)C2(CC2)C1 C12(NC(COc3cc(C)cc(C)c3)=O)CCC(C(=O)NC3CCOC3=O)(CC1)CC2 C1(C(=O)NCC2CCC(C)N(C(=O)C=C(Cl)Cl)C2)Cc2ccccc2N1 N1(C(c2ccnc(F)c2F)=O)CC2CCCN(C(=O)C3=CCCS3)C2C1 CCC(C)C(O)C(=O)N(c1cn[nH]c1)CCC1CC(C)N(C(c2cc(C)no2)=O)C1 C12(NC(=O)CNC(c3ncc[nH]3)=O)CCC(CC1NC(C1CCS(=O)(=O)N1)=O)C2 N1(C(C(CC)OC)=O)CCN(C(=O)Cc2cnsc2)C(C(C)C)C1 N#CC1(C(=O)NCC2CC(NC(C3CCCNC3=O)=O)CCO2)CC=CC1 c1(CC(=O)NC(CNC(c2c(CCC)occ2)=O)C)csc2sc(CC)cc12 C1(=CC(=O)NCC(CNC(CCCC(C)O)=O)O)CC2CCC(C1)N2C CCCCC(C(=O)N(CCCCCNC(C1OCCN(C)C1=O)=O)C)C(C)C N1(C(C(C)O)=O)CCCC12CCN(C(=O)CCC(=O)c1ccccc1Br)C2 C(CNC(c1onc(Br)c1C)=O)(C(C)C(C)C)NC(C(CC)=CC)=O c1(C(=O)NCCC2CN(C(C3C(C)CCC3)=O)C2)cc(F)cnc1O N1(C(C(C)S(C)(=O)=O)=O)CCCC(C2CCCN(C(C3COC(=O)N3C)=O)C2)C1 C(N=c1[nH]c(NCCCC2CCCN2C)nc2cccnc12)c1ccc(N)cc1 C1(CCNC(c2c[nH]nc2C2CCOC2)=O)CCCCN1C(C1CC(O)C1)=O c1(NC(=O)C(C)(C)C)ccc(-c2cn(CCC3CN(C(C)=O)C3)nn2)cc1 C1(C(=O)NC(c2nnnn2C)C)CN(C(C2CCC(C)(C)C2)=O)CC1F CC(C)C(C)CC(=O)N1CCN(C)CC1CNC(=O)CNc1cn(C)ccc1=O C(=O)(C1CCc2c(Cl)cccc21)N1CCC(C(=O)NC(COC)CO)CC1 Cc1noc2ncc(C(=O)OCCc3cnn(C)c3C)cc12 C(=O)(C1=C(F)CN(C(c2ncc[nH]2)=O)CC1)NC(C)(C)CC(F)(F)F N1(C(CCc2c(C)n[nH]c2C)=O)CCN(C(c2nn(C(F)F)cc2Cl)=O)CC(O)C1 c1(CC)onc(C)c1C(=O)NC(CC)C(=O)NCC(C)O c1(C(N(C2CC(NC(C3(F)CCCOC3)=O)C2)C)=O)cncc(F)c1Cl c1(NC(c2nc(-c3cccnc3-c3ccccc3)cs2)=O)cc(F)c(F)c(F)c1 C(CCCC(=O)NCc1ccc(C(=O)NC2(C(N)=O)CCOCC2)cc1)SC c1(OC)cc(CC(=O)NC2(CNC(c3nccc(Cl)c3F)=O)CC2)ccc1C Cc1csc(=O)n1CC(N1CCCC(C2CCCCN2C(c2cnn[nH]2)=O)C1)=O O=C1NC2CN(C(=O)CCC3CCN(C(C4CC4c4cccnc4)=O)C3)CC2O1 Cc1ccc(C(N2CCC(C(=O)O)CC2C)=O)c(CC(C)C)c1 O=C(C#CC1CCOC1)NC1CC(CNC(C2CC2C(F)F)=O)C1 CN1CC2CC1CN2C(=O)C(CCF)NC(c1cc2c(s1)CSC2)=O c1(O)ccc(N=[N+]=[N-])cc1.N1(C(CCC(C)NC(=O)C2CC2)=O)CCC(O)(C)C1 c1(C(N2CCN(C(c3c(C)coc3)=O)C(C(C)C)C2)=O)csc(=NC2CC2)[nH]1 Nc1cc(N2CCS(=O)CC2)ccc1C(=O)NC1CC1c1ccc(Br)s1 C(=O)(C(O)CCCc1ccccc1)NCCC1CC(NC(CNC(CC)=O)=O)C1 C12(C(=O)NCC(CCCC)NC(c3cc(Cl)ns3)=O)CC(CO)(C1)OC2C CC1(O)CON(C(=O)c2cc(C3CCCCC3)[nH]n2)C1 C12(CCC)C(=CC=CNN(CCC)CCC1)C(=O)NC(=O)C=CC2 c1(C(=O)NCC2(O)CC(CNC(=O)CCC3CCC3)C2)cnn2ccccc12 c1(N2CCC(OC(C)(C)C)C2)nc(SCCO)nc(C2CCCCC2)n1 c1(C(N2CC=C(CNC(C3C(CC)OCC3)=O)CC2)=O)cc(C)c(Cl)cc1C CCC(C(=O)NCC1(C)CCCN1C(c1cc(N)ccc1C)=O)C(C)C CCC(CNC(=O)C(=O)NCCCc1ccccc1)C(=O)O c1(CC(=O)NCC2(O)CN(C(CNC(=O)OC)=O)C2)ccc(CO)c(C)c1 C1(F)(C(N2CCC(CN(C(c3ccn(CC)n3)=O)C)C2)=O)CCOC1C N1(C(c2ncc(SC)nc2)=O)CC(C(=O)NCC(O)COC(C)C)CC1(C)C Cc1ccc(C(=O)NC2(CCNC(c3ccc(C4CC4)o3)=O)CCC2)cc1F Cc1cc(N2CCSCC2)ccc1NC(C1(C)COCCO1)=O N1(C(CC=CC)=O)CCCC(C2CCN(C(=O)C(C(C)C)SCC)CC2)CC1 c1(CNC(=O)CC2CCCN2C(=O)Cc2ccccn2)ccc(C(F)(F)F)cn1 c1(C(=O)NCCC(C)NC(C(CCC)C)=O)nn(C)c2ccc(Br)cc12 CCC(CC)CC(=O)NC(C1CCN(C(c2cc(C)n(CC)c2C)=O)CC1)C C1(C(N2CCC(CNC(=O)Cc3ccn(C(F)F)n3)CC2)=O)CCC(C2CC2)C1 CC(CN1CCN(C)CC1)CN=c1cc[nH]cc1S(=O)(=O)NC1CC2(CCC2)C1 Cc1c(C(=O)N(C(C)CNC(=O)Cc2cc(Br)cs2)C)cnn1C1CC1 CCC(C)(C)CC(=O)NCC1(F)CN(C(=O)C(C)COc2ccccc2)C1 CCCC(CC)C(=O)NC1CC1NC(c1ccc(C(C)=O)cc1)=O CN1CCN(C(c2cnc(-c3cnn(C)c3)cn2)=O)C(C#N)C1 C(=O)(CCC1=CCCCC1)N1CC(C)(CO)C(O)CC1.C12CC13CCN(C3)C2=O C1(n2cc(C3(C)CCN(C(C4CCOC4C=C)=O)C3)nn2)(CC=C)CCOCC1 Cc1c(Cl)sc(Cl)c1C(=O)NC(C)CCN(C(=O)C(O)CC1CC1)C c1(C(N2C(C(=O)Nc3c(C(N)=O)cccn3)CC2)=O)ccc(Cl)cc1Br C(C)(c1ccco1)=CC(N1C(C)(CC(=O)NC(C#C)C(C)OC)CC1)=O c1(NC(C2N(C(C)=O)CSC2)=O)cccc(NC(=O)CN(CCO)CCO)c1 C#CC1(O)CCCN(C(=O)C(c2cccnc2)NC(C23CCCCC2C3)=O)C1 c12cccc(c1)NC2=O.C(CF)(CF)(CO)NCCCOc1ccccn1 N1(C(CC(C(C)C)C)=O)CC(C)CN(C(c2cc3c(nc2O)CCC3)=O)CC1C c1(N(C)C)cncc(C(=O)NC2CCN(C(C3CCCN3C(N)=O)=O)CC2)c1 C1(CC)CCCC(NC(=O)C(Cc2ccoc2)NC(c2cnnc(C)c2)=O)C1 C1(NC(C(F)=CC)=O)COCC1NC(c1scnc1CC)=O N1(C(c2cnn(CCC)c2C)C(=O)NC(C)C)CCNC(=O)C(F)(F)C1 Cc1cc(Cl)cc(C(N2CC3(C2)CN(C(=O)Cc2ccc(C#N)cc2)C3)=O)c1C c1(C(N(CCN(C(C=NOC)=O)C)C(C)C)=O)cnc2c(C)cc(C)cn12 C=CC(CC)CC(=O)N1CCN(C(c2cc(Br)cnc2C)=O)C(CC)C1 C(C(CC1CC1)C(=O)NCC1(c2ccco2)CC1)NC(COCC)=O C1(CNC(c2c(C)ncs2)=O)C2CC1N(C(c1nn(C)cc1Cl)=O)C2 C1(CC(=O)NC2CN(C(c3coc(CO)c3)=O)C2)CCN(CC(F)(F)F)CC1 C1(NC(C2(C(=O)OC)CCCC2)=O)CC2(C1)CC(NC(=O)C(O)c1cnc[nH]1)C2 C(=O)(NNc1ccc(Cl)cc1F)c1cccc(CC=C)c1 C1(NC(N(CC)CC)=O)CC2(C1)C(C(=O)OC)C2(F)F.c1cc(C)c[nH]1 N1(C(Cn2ncc(C)c2)=O)CC(NC(c2nn(C)cc2N)=O)CC12CCOCC2 N1(C(c2ncn(C(C)C)c2)=O)CC2CC(C(N3CC(C)(C)C3)=O)(C2)C1 N1(C(C2(OC)CCC2)=O)CC(NC(c2ccc(C3(F)COC3)cc2)=O)C(C)C1 C=CC1(CC(=O)NCCn2ccnc2CO)CN(C(C2(CN3CCCC3)CC2)=O)C1 C(C(C(C)(C)C)NC(c1ccnn1C1CCC1)=O)NC(CC=CC=C)=O c1(C(N2CCN(C(c3c(C)nco3)=O)CC2CF)=O)ccc2c(c1)nnn2C O=S(=O)(c1cc(Cl)cc(Br)c1)NCc1cccc2nc[nH]c12 Cc1ccc(C(=O)CCC=O)cc1C.N1(C=O)CCCC(C(C)N)C1 C(=O)(CC(F)(F)CC)NC1(C(=O)NC(CC#C)CO)CCSC1 c1(C(=O)NCC(CCNC(c2ccc(C#N)s2)=O)O)ccc2cnccc2c1 C1(CSC)CC2(C1)CN(C(=O)C(C(C)C)OCC(C)C)C2.C1C(=O)N1 Cc1cc(C(N2CCCCC2C(C)NC(C2(C)CCC2)=O)=O)nn1C(C)C1CC1 N1(C(CC(C)(C)N(C(C)=O)C)=O)CCCC(C)C1CCO.c1(C2CC2)cccnc1 C(C(=O)NC(Cn1cncn1)C(=O)NCC(c1nncn1C)C)(C(C)C)OCC N1(C(c2nn(C)c(C3CC3)c2)=O)CCC(CO)C(NC(c2cccc(F)c2)=O)C1 CC(C(=O)NCC(O)C(=O)NCC1CCCC1(C)C)C(F)F c1(C(N2CC(C(C)NC(c3ccn(CCC)n3)=O)C2)=O)cccc2c1OCC2 n1(CC(=O)NCC2C3CN(C(c4cccc(CO)c4)=O)CC23)cnc([N+](=O)[O-])n1 C1(CN(C(C(F)=CC)=O)CC)CCCCN1C(c1ccc(C2CCOC2)cc1)=O c1(CC)nc(O)c(C(N2CCN(C(=O)CC3CC(F)C3)CC(O)C2)=O)cc1C CCC(CS(C)(=O)=O)N=c1nc2c(cnn2C)c(NCCOCC2CCOC2)[nH]1 C1(C(=O)NCC(CCOC)NC(=O)COc2ccc(C)cc2)CCC12CCC2 c1(NC(c2c(C)cc(CNC(=O)CCc3ccccn3)o2)=O)cccc(Cl)c1C C(=O)(CC(CC)CCCC)NC(CC=C)C(=O)NC1COCC(C)O1 c1(C(=O)NC(C2CCN(C(CC3(C(=O)OC)CC3)=O)C2)C)c(OC)ccnc1F Cc1ccnc(C(=O)NCC(O)CN(C)C(c2cc(N(C)C)ccn2)=O)n1 c1(C(N)=O)ccccc1C(=O)Oc1cccc(C(N2CCCC(O)C2)=O)c1 C1(CN(C)C)CN(C(=O)C(C)(C)C#N)CCO1.C(=O)(C(F)(F)c1cnccn1)NCC Cc1ccc(C(F)(F)C(=O)NCC(O)CNC(c2cc(C)[nH]c2C)=O)cc1 C=CC1(C(=O)N(C)CC2COC(=O)N2)CCN(C(c2cc(C)co2)=O)C1 CON1CCC(C(=O)NC2CC3CN(C(C4CCCC(=O)N4C)=O)CC23)CC1 c1(C(CC(=O)N2CC(n3cc(C4CCCCO4)nn3)C2)C(=O)O)ccc(Br)cc1 N1(C(C(c2ccc(C)s2)C)=O)CC(O)C(O)C1CNC(C1(C)CCN(C)CC1)=O C1(CCC(=O)NCCN(C(C)C)C(C)C)(NC(C2CC(SC)C2)=O)CCCC1 C1(NC(C(C)(O)CC(=O)c2ccccc2)=O)C2COCC1CN(C(=O)C1CC1)C2 CC(C(=O)NC1CC2CC1N(C(=O)Cn1c(C)csc1=O)C2)S(N)(=O)=O C1(CC)(NC(C2CC(NC(=O)CN=[N+]=[N-])C2(C)C)=O)CCCCCC1 C(=O)(C#CC1CCOC1)NCCCN(C(C1N(C(C)=O)CCCC1)=O)C c1(C(=O)NC2C(NC(C(S(C(C)C)(=O)=O)C)=O)C2)c[nH]c2c(Cl)cccc2c1=O C1(C(=O)NCCc2c(OC)cccc2)CN(C(C2CC(C)N(C)C2)=O)CC1(C)C C1(OC)CC(C(=O)N(C2CCCC2C#N)C)N(C(=O)C(C)SC(C)C)C1 c1(C(CNC(C2SC3C=CC2CC3)=O)NC(CCC=C)=O)cc(F)cc(Cl)c1 C=C(Cl)CC(C(=O)N1CC2CC2(CO)C1)NC(=O)CCC1CCOCC1 N1(Cc2scc(C)n2)CCc2sc(-c3cccc4c3CC(=O)N4)nc2C1 N1(C2CC(CNC(C3(C)CC3(Cl)Cl)=O)C2)CCC(NC(c2cc(C#N)c[nH]2)=O)CC1 Cc1ccc(CC(=O)NC2CCCN(C(c3c[nH]c(Br)c3)=O)C2C)cc1O N1(C(c2cc(C)ns2)=O)CC(C(=O)NC2CC2c2ccnn2C)CC12CCC2 C(=O)(C(CC(C)C)ONC(=O)C(CN(C)C)N(C)C)NCc1c(C)nccn1 c1(C(=O)NCC(C)CNC(=O)C(c2ccc(F)cc2)(C)O)cccc2cnsc12 C(C1(C)CCOCC1)=CC(=O)NCC(CC)NC(=O)CC1(c2ccon2)CC1 C12(CC(=O)OCC)CCNC1CN(C(=O)NCCOCC1CCCO1)C2 CCCC(C)C(=O)NCc1ccc(C(=O)NC2CC(C)(C(N)=O)C2)nc1 C(=O)(C(O)CC(F)(F)F)N(C)CC1CCN(C(=O)CSc2ccccc2)CC1 N1(C(CCOC)=O)CCCC(C)(CNC(=O)CCn2nc(C)nc2C)C1 c1(OC)cc(C(N2CCC(c3cn(C4CC4)nn3)CC2C)=O)ccc1C#N c1(CN2CCCN(C(C(C3CCCN(CC)C3)(C)C)=O)CC2)ccc(F)cc1F C(=O)(C(O)C(C)(C)CC)N1C(CNC(c2ccc(C#C)cn2)=O)CC(C)(C)C1 C1(NC(c2c(SC)ccs2)=O)CN(C(=O)Cc2conc2C)CC2(CC2)C1 c1(NC(C2(F)CCN(C(c3c(C)ncnc3)=O)C2)=O)ccc(C(F)(F)F)c(C#N)c1 C1(c2ccccc2)(NC(=O)CSC(F)F)CCN(C(C2CCC2)=O)C1 c1(C(=O)NCC#CCNC(C2(O)CCC(CC)C2)=O)ncc(N)cc1Cl Cc1cnc(C)c(C(N2CCCC(CN(C)C(c3cc4n(n3)CCO4)=O)C2)=O)c1 c1(N2CCC(NC(CC)=O)C(C)(C)C2)nc2cc(F)ccc2o1 C(=O)(C1CCCn2c(C)cnc21)N1C(CC)CN(C(=O)CCN(C)CCO)CC1 N1(C(C(CC#C)C)=O)CCCCC(CNC(=O)CCC(=O)c2ccncc2)C1 N1(C(CN(C(C)=O)C)=O)CCC(CC(=O)NC(C)C(C)n2cncn2)(O)C1 C(=O)(C#CC1CCCO1)NC1(CCC)CCN(C(=O)CC(CC)OCC)CC1 C(C(CC(C)C)C(=O)N1CCC(N(C(=O)C(CC)(CC)CO)C)C1)OC C1CCCC(=O)N(S(C)(=O)=O)CCc2cn1nn2.CC(C)C(F)NCCO CC1(C)CCC12NC(=O)N(C1CCCN(C(c3ccc(Cl)cc3)=O)CC1)C2=O c1(C(=O)NCC(O)C(=O)NCCCc2ncco2)coc2ccccc12 N1(C(C(C(C)C)NC=O)=O)CC2(C=C(C(=O)NCC3CCCC3C)CO2)C1 c1(CC(=O)NCC(CN(C(=O)COc2ccc(F)cc2)C)O)nc([N+](=O)[O-])n[nH]1 Cc1nc(NC(C)C(C2CCCCC2)NC(c2cocc2C)=O)c2ccsc2n1 C(=O)(CC1OCCc2ccccc21)NC1(CN(C(c2nc(C)oc2C)=O)C)CC1 C(CC(C(C)(C)C)NC(=O)CC(CC)CC)N(C(C(CC)N(C)C)=O)C C(=O)(C(F)(F)C(F)(F)C(F)F)NC1C(NC(c2c(CSC)cccn2)=O)C1 C(=O)(CCCCCC(CC)NC(=O)OC(C)(C)C)NCCN(C(C(C=C)O)=O)CC C1(CN2CCC(NC(C(C)NS(CC)(=O)=O)=O)C2)CCC(CO)CC1 N1(C(c2ccc(OC)c(OC)c2)=O)CCC2(CC1)CCN(C(C1CC(C)C1)=O)C2 c1(C2CCN(C(=O)NCC(c3cccc(C)c3)C)C2C)ccc(C#N)cc1 c1(C(=O)NC2C(CNC(c3c(C)c(F)ccc3)=O)C2)ccc2c(c1)N(C)CC2 c1(OCCC2CCCC2)ccc(C)c(-c2cc(C(=O)N)n[nH]2)c1.c1(COC)ccccc1 C(=O)(CCC(=O)NC1CCCC(N(C(=O)CC(C)(C)C2CC2)C)C1)N(C)C C1(C(=O)NCc2c(C(N(CCCC)CC)=O)n(C)nn2)CCCC(C)(C)C1 C1(CNC(COCCC#C)=O)COCCN1C(=O)C(c1ccc(Cl)cc1)CC S(=O)(=O)(c1ccc(C#N)c(NC(C)CS(C)(=O)=O)c1)NCCCN(C(C)C)C c1(C(=O)NC(C)C(F)(F)C(F)(F)F)ccc2c(c1)CCC2N C=CCC(C)(C)C(=O)NC1C2CC3C1C3C2C(N1CCCC1Cn1ccnc1)=O c1(C(N(CC(F)(F)F)CCN(C(COc2ccccc2)=O)C)=O)ccc(OC)cc1 c1(Nc2ncn(C(C)C)n2)ccc(C)cc1.C1(C(=O)N)CC(N)C1(C)C C1(CC)CN(C(=O)C(O)CNC(c2ccc(OC)nc2)=O)CCN1C c1(C(=O)NCCC(C)(C)NC(Cn2ncc(C)c2)=O)ccc2ccccc2c1O N1(C(C2(C(=O)OC)CC2)=O)CCc2ccccc2C1CCNC(=O)C(OC)OC N1(C(CCN)=O)CCc2nc[nH]c2C1.C1(CC(=O)CC#C)CCCC1C C1(C(=O)NC2CC(C)N(C(C3CC(C)(O)C3)=O)CC2)CCc2ccccc2CC1 c12cccnc1N1CC=CC(C1)COC2=O.C1(C(=O)NCC)CC=CCO1 N1(CC)C(=O)CCC1C(=O)NC(C1CCN(C(c2csnc2C)=O)CC1)C N1(C(C=COCC)=O)CCC(O)(CCNC(C2CCCCC2C(N)=O)=O)C1 C(=O)(C(F)(F)C(C)(C)O)NCCCCN(C)C(c1cccc(F)c1Cl)=O c1(C(=O)Nc2ccc(N3CCN(S(=O)(=O)C(F)(F)F)CC3)nc2)csc2ccccc12 C12(C(N(CCN(C(=O)COCC3CCOC3)C)C)=O)CCN(CC1)CC2 c1(C(=O)NCCCCC(C)NC(=O)CN2CCCCC2)coc2c1C(=O)CCC2 C(N=c1ccnc(C)[nH]1)C12CC(NC(C(C)OCC)=O)(C1)C2 CC1(NC(=O)CC(O)CNC(C2CCCCO2)=O)CC2(CCC2)C1 CC(C)(CCC#N)C(=O)NCc1cc(C(N2CCSC3CCCC23)=O)no1 C12C(CCCC1C)NC(=O)N2.C1(OC)COCC1N1CCCC1 N1(C(C(C)SCC)=O)CCC(COC)(NC(c2conc2CC(C)C)=O)C1 c1(C(=O)Nc2scc(-c3scc(C(=O)NC(CC)CC)c3)n2)cc(C)cc(C)c1 c1(-c2ccc(C(=O)NC(C(C)(C3CC3)OC)C)s2)ccc(F)cc1F C1(CNC(C2C(C)OCCO2)=O)CN(C(=O)C(=O)Nc2ccccc2)CC1(C)C CC1CC(C(N2CCC(C(=O)ON)C2)=O)CN(C(=O)CCNC(=O)OC(C)(C)C)C1 c1(C(CC)C(=O)NC(C)CNC(c2cc(C)cs2)=O)ccc(F)cc1 N1(C(CC(=O)NCC)=O)CCCCC1C(=O)NCC1(CC)CCCCC1 C1(C(=O)NC(CC=C)C)CC2(CC2)CN1C(=O)C=Cc1ccnn1C C1(C(N2CCCC(CCCC)C2)=O)CN(C(=O)CNC=O)CC1C1CC1 N1(C(c2c(C)cns2)=O)CC=C(C(C)(C)C(=O)N2CCCC(C)(C#N)C2)C1 c1(OC)c(C(=O)NC2CC3CCC2N(C(=O)CO)C3)cnc2ccccc12 c1(C(=O)NCC2CN(C(C3(C)CCCS3(=O)=O)=O)CC2O)cnn2ncccc12 CCCCCC(=O)NCC(C)(CNC(C1CCN(CC)C1)=O)OC C(=O)(CCCC(=O)NOC(C)(C)C)NCC1N(C(C(OC)OC)=O)CC=C1 c1(OC)ccc2c(c1)C(C(=O)N1CCC3(C1)CN(C(=O)C(C)=C1CC1)C3)CCC2 Cn1cnc2sc(C(=O)NC3CC(CNC(=O)Cc4cnc[nH]4)C34CCC4)cc12 CC1CCN(C(=O)CC2CC(C)(C)CCO2)CC1N(C(=O)CCC(F)F)C C#CCCCC(C)(c1nnnn1C(C)C)NCC(CO)C(F)(F)F N#Cc1cccc2[nH]cc(C(=O)NCC3CCN3C(c3cn4c(n3)SCC4)=O)c12 c1(Cc2c(OC)ncnc2N2CCCC3(COC3)C2)n[nH]c2ccccc12 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC1CC(N(C(=O)CSC(F)(F)F)CC)C1 O=S(=O)(c1ccc(N2C3CCC2CC(O)C3)c(F)c1)NCCc1ccno1 N1(C(CC2CCN(C)C2=O)=O)CC2CC(C1)CN(C(C1(CO)CC(F)(F)C1)=O)C2 N1(C(C)C(=O)N(CCO)CCN(C)C)CC(C)(C)CC1C(=O)Nc1ncccc1F N1(C(C2(C#C)CCC2)=O)CC=C(CC(=O)NCc2cc(O)ns2)CC1 N1(C(CN(C)C)=O)CC(C)(C)C(NC(=O)CCF)C(C)(C)C1 C1(C(N2CCC(CNC(C3CC4C=CC3C4)=O)C2)=O)(CC)CCNC1=O C1(c2ccc(CC)cc2)CN(C(=O)CSC(C)C)CCN1C(=O)Cn1cnnn1 C1(NC(Cc2cnc(C)s2)=O)CC2(C1)CN(C(=O)Cc1cccs1)C2 C=CCC(C(=O)N1CCCC1CNC(=O)CSc1ccc(OC)cc1)NC(C)=O CCC(C)CC(C)N(C)C(C1(NC(c2cnn(C)c2C)=O)CC1C)=O C(=O)(CC(C)C(F)(F)F)N(C(C(NOC(C)CC(F)(F)F)=O)C)C c1(COC(=O)Cc2ccn(CSc3ccccc3)n2)c(F)cncc1F N1(C(C2(NC)CC2)=O)CC(OC)CC1C(=O)NCc1nnn(C)c1C n1(CCN(C(CC(=O)NC)C2CCOCC2)CCOC)cc([N+](=O)[O-])cn1 c1(C(N(CC(C)(C)CNC(=O)CC2(C)CC2(F)Cl)C)=O)[nH]nc2ncccc12 C(=O)(C=C1SCC(=O)N1C)NC1CC2(CN(C(C(C=C)(C)CCOC)=O)C2)OC1 c1(C(N(C(CNC(=O)CN2CCS(=O)CC2)C2CC2)C)=O)cnn2c1CCCC2 C1(NC(C2(CC=C)CCN(C(C3C(C)C3C)=O)C2)=O)CCCC(O)CC1 C1(NC(=O)COCC2CC2)CN(C(c2c(F)ccc(O)c2F)=O)CCC12CCC2 c1(C(=O)Nc2c(NCc3cccc(OC)n3)ccs2)c(Br)cc(Br)c(C)c1Br N1(C(C2(C(=O)OC)CC2)=O)CCCC(O)(CNC(=O)C(C)c2cccs2)C1 C(C(C)(C)C(N)=O)NC(C1N(C(C2C(CC)N(C)CC2)=O)C(C2CC2)CC1)=O c1(C(=O)NC2C(NC(CC(CCC)C)=O)CC2)cn(CCO)c(=O)nc1O C1(COC)CN(C(C2CN(C(C3(SC)CC(=O)C3)=O)CC2F)=O)CCO1 C(=O)(CCCS(C)(=O)=O)NCCOCCCNC(c1c(C#C)c[nH]n1)=O c1(C(N(C)CC2OCCN(C(C(C)C(C)(F)F)=O)C2)=O)cc(S(N)(=O)=O)oc1Cl c1(C(N2CC(O)(CN(C(c3nn(CC)c(C)c3)=O)C)C2)=O)cc(OC)ccc1F C1(C)(C(N(CC(C)N(C)C(c2occc2C2CC2)=O)C)=O)CCN(C)C1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)COCC2CCC2)CCC12CCOCC2 C1(NC(C(C)N(C)Cc2cc(Cl)cc(Cl)c2)=O)CNc2ccccc2C1 c1(C(=O)NCCC2OCCCN(C(CC(C=C)C)=O)C2)nn(C)c2ccccc12 c1(C(=O)NC2CCC(NC(C3CCN(C)CC3)=O)CC2)ccc([N+](=O)[O-])c(Cl)c1 C(=O)(CC(C)(C)n1cc(CC(c2ccccn2)O)nn1)NC(CC=C)C C1(NC(COCCOCC)=O)CN(C(C2(N=[N+]=[N-])CC2)=O)CC1(C)C C1(CNC(c2c(C(C)C)nns2)=O)CCCN(C(c2cnc(S)n2C2CC2)=O)C1 C1(NC(=O)CCc2ccnc(C(F)(F)F)c2)C2Cc3c(Br)cccc3C12 C(=O)(C(C)CCC(C)(C)C)N(C1CCN(C(C)C(=O)OC)C1)C1CC(F)(F)C1 c1(C(=O)NC(CNC(C(CCC)OC)=O)C(C)C)cc2c(C)cccn2n1 C1(NC(c2c(C(C)C)scn2)=O)CN(C(c2cc(Cl)on2)=O)CC2(CCC2)C1 C1(C(=O)NCCc2n(C)cnc2)N(C(=O)CN2CCC(F)CC2)CC12CCCC2 c1(C(=O)NC2(CCNC(=O)C3=CCOC3)CCC2)ccc(=O)n(CC(F)(F)F)n1 Cc1nc(C(=O)NC(C(C)NC(c2ncoc2-c2ccsc2)=O)C(C)C)c(C)s1 CC1OC2CCC1(C(=O)NCCC1(NC(=O)CCCCCN(C)C)CCC1)C2 C#CCC(CC#C)C(=O)N1CCC(CCNC(C2(C3CC3)CCC2)=O)C1 N=c1cc[nH]c(C(N2CC3C(CC(=O)NCCCN=[N+]=[N-])C3C2)=O)n1 Cc1cccc(C(=O)NCCN2CCCN(C(=O)C3=C(Cl)CC3)CC2)c1O C1(NC(C(CCC)c2ccccc2)=O)CC2CCC1N2C(=O)C(=O)N(C)C c1(C(C)N(C(C(=O)Nc2ccccc2)c2cc[nH]n2)C)cn(C)cn1 CC(C)CCCC(C)CNC(=O)C(C)(CO)NC(=O)CC1(O)CCCCC1 C1(OCC)CCC(N(S(=O)(=O)CCCOC(C)(C)C)C)CC1 C1(NC(C(CC2CC2)OC)=O)CN(C(c2ccc(C)cc2)=O)CC2(CCC2)C1 C1(C(NOC(C(=O)OC)C)=O)OCCC1NC(=O)C=C(C)C(C)(C)C CC1(C)SCC=C1C(C(=O)NCC1CC2(CCOCC2)CO1)N1CCNC(=O)C1 c1(C(=O)NCC2(COC)CN(C(C3CCC3C)=O)C2)nccc(C)c1Br N12CC(N=C3C=CN=C(N3)C1)C2.c1(OCCC(=O)OC)ccccc1OC CC1=C(C(=O)N2CC(CCCCNC(c3csc(C(F)F)n3)=O)C2)CCCO1 n1(CC(=C)C)nnnc1C1(NC2CC(C(N)=O)C2)CC(C(C)C)C1 c1(C(N2CC(CN(C(C=CCC)=O)C)OCC2)=O)cc2c(C)cc(Cl)cc2[nH]1 c1(C(N(C)CC2CCN(C(C3(C#C)CC3)=O)CC2)=O)c(C)[nH]c2ccccc12 C1(NC(CCOCC#C)=O)CCCN(C(=O)C(C)Oc2ccc(Cl)cc2)C1 c1(NC(C)Cc2ccc(Br)cc2F)ccc2[nH]c(C(=O)O)cc2c1 C(=O)(C(C)S(N)(=O)=O)NCCC(C(=O)NC(c1ccccc1)C)OC N1(CC(C(=O)C(N2CCCC(O)C2)C)=O)CCOC(C)(CN(C(CC)(C)C)OC)C1 N1(C(c2c(C)nncc2)=O)C2CCC1CC(NC(C1(C)CC1(F)F)=O)C2 C1(NCC(c2ccc(F)cc2F)(C)OC)CS(=O)(=O)CC1C c1(CCC(C(=O)NCC(=C)C)N2CCC(C(=O)NC)CC2)ccnc(F)c1 N1(C(C(c2cn(C)nn2)N(C)CC2CC2)=O)CCCC1CC1CCCO1 c1(-c2cccc(C#C)c2)cnn2cc(C(=O)Nc3ccc(C(C)O)cc3)cnc12 c1(OC(C)=O)cccc(CNc2c[nH]nc2C(=O)NCC(O)CO)c1 C1(C)(C(N(CCC)CCNC(=O)CC(CSC)OC)=O)CCOC(C)C1 c1(C(N2C(C)CC(CNC(C=CSC)=O)C2)=O)ccc(O)nc1Cl N1(C(C(CC=C)C)=O)CCCC(NC(=O)C(CC)c2cccnc2)CC1 Cn1cnc2cncc(C(=O)NCC3(F)CCN(C(=O)CCS(C)(=O)=O)C3)c12 N1(C(CC(=O)OC)=O)CCCC1C=CC(=O)N(C)Cc1cn(C)nc1C N1(C(c2ccc(COC)s2)=O)CC2(NC(c3ccccc3C)=O)CC1C2 c1(C(N2CCC(NC(C(CCSC)O)=O)C2C2CC2)=O)cc(F)ccc1O C(C(C)(C)CNC(=O)CCOC1CN(C(=O)CCn2cnc(=N)[nH]2)C1)OC CC1OC(C)CC1C(=O)NCC(O)CNC(c1snnc1C1CC1)=O c1(C(N(C)CC2(C(N3CCCC3)=O)CC2)=O)cc(C#N)no1.C(=O)(CN)NC C1(CNC(C(c2ccccc2)OC)=O)CC(F)CN1C(C1CCC(C)C1)=O N1(C(c2ccc(C(CC)(C)C)cc2)=O)CC(C#N)N2CCC1C2 C=CC1(CC(=O)NC2CCN(C(C3CC(OC)C3)=O)CC2F)CCCCC1 N1(C(c2cccc(OC)n2)=O)CCC2(C1)CN(C(=O)CCOC(C)C)CCO2 c1(C(N2CC3CC(F)(C3)C2)=O)c[nH]c2cc(F)cc(F)c12 C1(CCCNC(C2(F)C(C)C2)=O)CCCCN1C(c1cccc(C2CC2)c1)=O C1(CNC(CC2C(C)(C)CCCO2)=O)C(C2CC2)CCN1Cc1ccccc1 C=CCC(C)(CC)C(=O)NC(C1CCN(C(=O)Cc2ccc(C)c(F)c2)CC1)C Cc1cccnc1C=CC(=O)NC1CC2CC(NC(C34CCCC3C4(F)F)=O)C1C2 C1(C(=O)NC2CCC(CC)C2)(CNC(C(C2CC2)OCC)=O)CCCC1 c1(C(N2CC(C(C)NC(CC=C)=O)C2)=O)cc(F)c(F)c(F)c1 Cc1nc2cccc(Cl)c2cc1C(=O)OC(c1ccccc1Br)C(F)(F)F C1(C(=O)NC(CCNC(COCC(C)C)=O)(C)C)Cc2ccccc2O1 c1(C(=O)NCC2COCCN2C(=O)Cc2ccc(Br)c(F)c2)cnc(O)cc1O Cc1cc(F)c(Cl)cc1C(=O)NC1CCN(C(=O)COCCC(C)C)C12CCC2 N12CCC(C)(CC1)C2.N1(C(C)=O)CC(OC(=O)N(C)C)C1 N1(C(C2N(C(c3c(CC)ncnc3)=O)CCC=C2)=O)CCCC(C)(C#N)C1 C#CCCCC(=O)NCC(C1CCN(C(C2(COC(C)C)CC2)=O)CC1)C C1(C(=O)NCc2c(C(=O)NC3CC(CC(C)(C)C)C3)occ2)CCC=CCCC1 c1(C(=O)NCCC(C)Nc2nc(OCC)c(Cl)cn2)cccc2nc(O)ccc12 C1(CNC(C2CC(OC)(OC)C2)=O)CC2CCC1N2C(=O)Cn1ccc(C)n1 CCC(C(=O)NC1(C)CC(NC(c2n[nH]c(C)c2Cl)=O)C1)C(F)(F)F Cc1cc(NC(=O)C(C)C(C)NC(=O)C(C)(C)CC#N)c(C)c(C)c1 C1(NC(C(CC(N)=O)O)=O)CN(C(c2cnccc2Cl)=O)Cc2ccnn2C1 Cc1cc(C(=O)NC2CC(N(C)C(c3cc4ncccn4n3)=O)C2)c(C)c(C)c1 C1(CNC(C2(CCCC)CCC2)=O)CCCCN(C(=O)CCC(C)(C)C)C1 N1(C(C(CO)OC)=O)CCC(C(=O)NC(C)Cc2ccccn2)C(O)C1 C12(c3nnc(-n4nc(C)c(C)c4C)o3)CCN(C(=O)CCC(C)C)CCC1C2 C(=O)(CCCCCCNC(=O)C(F)C(C)C)N(CCC(=O)OCC)C c1(C(=O)NCCN(C)C(C2CC3(CCC3O)C2)=O)cc2c(c([N+](=O)[O-])c1)OCO2 C12(NC(=O)CCc3nc[nH]n3)CCC(CC1NC(=O)CN1CCNC1=O)C2 C(=O)(C1CC(=O)Nc2ccccc21)NC1(CO)CN(C(CNS(CC)(=O)=O)=O)C1 C(=O)(C(C)(C)CC(F)F)NC(CC)CCC(=O)NC(CO)CC(F)(F)F C1(CNC(C(C)OCC(F)(F)F)=O)COCCN1C(c1cc(C(C)(C)C)on1)=O n1(CC(=O)N(C(C)C)CCNC(C2C(Cl)(Cl)C23CC3)=O)nc2n(c1=O)CCCC2 c1(C(=O)NCC2(NC(c3n(C)nc(O)c3)=O)CC2)ccnc(F)c1N C12(C(=O)NC(C3CCN(C(c4c(C)csc4)=O)C3)C)CC(CN1C1CC1)C2 c1(OC)cncc(C(N2CC(O)(CCNC(=O)CC3CCN(C)C3=O)C2)=O)c1 n1(CC)c(C(=O)N(CC(C)C(=O)N2CC(F)(C(=O)OC)C2)C)cnc1O c1(N2CCC(CN(C(=O)CCC(C)C)CC#C)CC2)nc(C)cc(C)c1C#N Cc1[nH]nc2ncnc(N3CCCC4(C(=O)NC5(C6CCCO6)CC5)CC4C3)c12 c1(C(=O)NCC(C)CNC(c2cccc(C(N)=O)n2)=O)cc2cc(Cl)ccn2n1 c1(C(=O)OC)cc(C)c(NC(c2nnn(-c3cccc(Cl)c3)c2C)=O)c(Br)c1 CC1(C)CCOC1C(=O)NC1CC(Cn2cc(CCSCC3CCCCO3)nn2)C1 c1(C(N2CC(C(C(=O)NCCN3CCCCC3)O)C2)=O)cc(O)cc(=O)o1 C=CC(C)(C)CC(=O)N1CCN(C(c2cnc(S)nc2)=O)C(CF)C1 C(C1CN(C(C2(F)CC2)=O)CC1C(=O)NC(CN1CCCC1)C(C)C)=CC c1(C(=O)NC2CN(C(C3CC(CF)C3)=O)C2)ccn(CC(F)(F)F)c(=O)c1 Cc1cc(C(=O)N(CCCN(C)C)CCNC(C2CCC(C)(C)C2)=O)cc(=O)n1C N1(C(C2(C=C)CC2)=O)CCN(CC2CN(C(=O)CCF)C2)CC1 C12(NC(CN(C)C)=O)CCCC1CN(C(c1cc(C(F)F)ccc1F)=O)C2 C1(CC)CCCCC1C(N1CC(O)(CNC(c2cc(C)ncn2)=O)C1)=O C1(OC(C2C(C)(C)CCCO2)=O)CCc2scnc2C1 c1(OCC)ccccc1CCC(N1CC2CC2(NC(=O)CCS(C)=O)C1)=O N1(C(c2cccc(C)n2)C(=O)NCCC2(C)CC2)CCc2cncnc2C1 C1(C(N(C2CC(NC(c3cccc(CS(C)=O)c3)=O)C2)C)=O)OCCC1(C)C c1(OC)cncc(C(=O)NCC(O)C(=O)N(CC(O)C2CC2)C)c1 N1(C(=O)NCC2CCCCS2(=O)=O)CCC(F)(F)C(CO)C1.C1CCCNC12CC2 N1(C(C2(CCC=C)CC2)=O)CCC(c2n[nH]cc2CNC(=O)CC(C)C)C1 c1(OCC)cc(CN2CCN(C(=O)CNC(=O)NC)CC2CC)cc(F)c1 C(=O)(C1=CCC(NC(=O)CN2CCCCC2C)C1)NC1(CCOC)CCC1 N1(C(c2c(C)nc(Br)cc2)=O)CC2(CCN(c3ncncc3C#N)CC2)C1 N1(C(c2n(C(CC)CC)ncc2)=O)CC2CCC1C(CNC(=O)CC(C)OC)C2 C(C(F)(F)CC(O)CO)N(C(=O)C(O)C1(NCCC(=O)O)CCC1)C C1(N(C)C)(CC)CCN(C(c2scnc2C)C(=O)Nc2cccc(F)c2)C1.C1CS1 N1(C(C2CC(C(=O)OC)C2)=O)CC(NC(C2CCCC(C)(C)O2)=O)C2(CCC2)C1 CCCN(OC)C(=O)C1(C(=O)OC)CCN(C2CCC(C)(C)OC2)C1 c1(C(=O)OC)cc(C(=O)NCC2CCCC2NC(C23CC(CO)(C2)C3)=O)n(C)n1 C1(NC(c2cc(OC)nn2C)=O)CC(F)CN(C(=O)Cc2ccsc2)C1 CC1=C(C(=O)N2CCC(C)C(NC(C3(C4CC4)CCC3)=O)C2)CCCO1 c1(C(=O)NCCC2(CNC(C3CC=CC3)=O)CC2)coc(CC2CCC2)n1 CCCCC(C)C(=O)N1CCCC(NC(=O)Cc2csc(C3CC3)n2)C1C c1(CC)cccc(CC(=O)NCC(CNC(=O)C(C)OCC2CC2)O)c1 CN=c1[nH]nc(CC(N2CC(CCNC(=O)COc3cn[nH]c3)C2)=O)s1 c1(C(N2CCN(C(c3c(CC)cccn3)=O)CC2CF)=O)ccnc2[nH]ncc12 CN1CC(NC(C2CSCCS2)=O)CC12CCC2 c1(C(N2C3CC(N(C(CC4C(C)C4)=O)C)CC2CC3)=O)ccc2[nH]c(=N)sc2c1 O=C(C1=CSCS1)NCC1CCN1C(=O)C(O)Cc1cnc[nH]1 C1(C(N(CC(=O)NCCC(F)(F)Cl)CCOC)=O)C2(CC2)C12CC2 c1(CC(=O)OC)cccc(C(=O)NCC23CC(CO)(C2)OC3C)c1 C(=O)(C(C)(C)C(C)SC)N1CCC(CNC(CN(C(=O)OC)C)=O)CC1.C(C)(C)(C)O N1(C(c2c(C)cc(C)s2)=O)CC(C(=O)NCC2(O)CCC(C)(C)C2)CC(C)(C)C1 c1(NC(C2N(Cc3c(C)cc(OC)c(C)c3)CC=C2)=O)cnc2ccccc2c1 C(=O)(C(C)(C)CC(=O)NC1CCN(C(C2CN(CC(C)C)C2)=O)CC1C)OC c1(N2CCC(C)C(NC(C(N3CCOCC3)C)=O)C2C)nc2ccc(F)cc2o1 CCC(CCOC)C(=O)NCC1CCCN1C(C1CC1(C)C)=O C1(C(N(C2CCN(C(c3coc(C)c3)=O)C2)CC(=O)OC)=O)CCCCC1 c1(C(N(CCOCCCN(C(C2C=C(C)CS2)=O)C)C)=O)ccc(F)cc1F N1(C(c2nc(CNC(C3(OCC)CCC3)=O)oc2)=O)CCC2CCC12 C1(CNC(c2cncc(C(F)(F)F)c2)=O)CN(C(c2ccccc2Cl)=O)C2CC12 c1(C(=O)NCCNC(c2nc(-c3ccc(C)o3)sc2)=O)cccc(C2(C)CC2)c1 C(=O)(C(F)(F)C(C)O)N1CCC(C(=O)NC(CCC)C)CC1 C12(C(=O)NC3C(NC(=O)CNC(=O)C4CC4)CCC3)CCC(CC1)CO2 N1(C(CCN2CCN(C)CC2)=O)CCC2(NC(c3nc(=O)n(C)[nH]3)=O)CCCC12 c1(C(N2CCC(Cc3ccccc3)C2)C(=O)NCCCF)ccc(F)c(CO)c1 c1(CC(=O)NCC2C(NC(c3ccn(CC)n3)=O)C2)ccc(Br)nc1 C1(C(N2CC(C)C(F)(F)C2)=O)CC(O)C(O)CC1CNC(C1CC(=O)N(C)C1)=O C1(C(C)(C)CNC(=O)CC2CC(C)(C)C2)CN(C(C2(F)CC=CCC2)=O)CCO1 C1(C(=O)NC2(CC=C)CCN(C(C3CCC(OC)CC3)=O)C2)CN(S(N)(=O)=O)C1 C1(NC(CCc2cc(C)no2)=O)CC2CCC1CN2C(=O)CC1(C)CCOCC1 Cc1cc(C(N2CC(NC(=O)CCOc3ccccc3F)C(C)C2)=O)ncc1F C1(c2cc(C(=O)OC)n[nH]2)CCN(N(C)C2CC3(CC=CC3)CC2)C1 CC(CC1CCCCC1)C(=O)NCCN(C(c1coc(Cl)n1)=O)C1CC1 c1(C(=O)NC2C(NC(CNC(CCC)=O)=O)CS(=O)(=O)C2)n[nH]c2ccccc12 CCC(CC(F)(F)F)C(=O)NC(C)CC(C)NC(=O)COc1ccc(C)cc1C Cc1sc(C(=O)NCCCCC2CCCN(C(C3C(C#N)C3(C)C)=O)C2)nc1O c1(C(=O)OCC(=O)Nc2ccc(C(C)=O)c(F)c2)cc2c(nn1)CCOC2 CC1(CNC(=O)C2=CSCS2)CCN(C(C2CC3CC3C2)=O)CC1 C(CC1CCOCC1)(C(=O)NCC1CC(C(N)=O)C1)NC(CCSCCCC)=O c1(N(C(CC2(C)CCCNS2(=O)=O)=O)CC2CCN2C(C)=O)c(F)ccc(N)c1F c1(CC)nc(C)c(C(=O)NCC2(O)CN(C(=O)CN3CCCC(N(C)C)C3)C2)s1 Nc1c(C(N2CCOC(CCNC(c3ccc(O)nc3)=O)C2)=O)ccc(Cl)c1F C1(CNC(C(CC)N(CC)CC)=O)CCCCN(C(c2cnn3c2CCC3)=O)C1 C1(CCNC(C2(OCC)CCC2)=O)C(C)CCCN1C(=O)CN(C)C c1(OC)ccnc(C(=O)NCC2CC(CNC(C3CC=CCO3)=O)C2)c1OC N1(C(=O)NCc2ccc(-n3ccnc3)nc2)C2CCC1C1CNCC21 c1(C(=O)NC(c2ccccc2)COC)cccc2cc(Br)cnc12 N1(C(Cc2nc(C)sc2)=O)CCCC(CN(C2CC2)Cc2ccsc2)C1 N1(C(c2c(OC)scc2)=O)CC2(CCC2NC(=O)Cc2cccc(F)c2Cl)C1 N1(C(CC2(OC)CC2)=O)CCCC2CN(C(=O)C(C)CC3CC3)CC12 CCC(C(=O)NCc1cn(CC(=O)N(C(C)C)Cc2cnc(C)s2)nn1)SC C#CC1(C(=O)NCC(C2CCCC2)NC(=O)C(F)(F)c2cnn(C)c2)CCCC1 C1(C(N(CCC(C)NC(=O)C2CC2)CC)=O)C2CCC1(c1ccc(F)cc1)C2 C(CCCCCCCO)NC(=NCCc1c(C)nn(C)c1)NCC1CCCS1 C1(C(N)=O)CN(C(=O)CCNC(C2CN3CCC2C3)=O)CC12CC2 c1(NC(=O)NCC2CCC(C)CN2C(=O)OC(C)(C)C)ccc2c(c1)CCO2 c1(C(=O)OC2CCCCC2)ccc(CN(C(CC2CCN(CC)C2)=O)CC)nc1 CC1(C)CC(NC(=O)CCc2cnco2)CN(C(c2ncoc2C2CC2)=O)C1 N1(C(=O)NC2C(C(=O)OCC)CCC2)CCCC2(C1)CN(C)C(=O)O2 N1(CC)CC2CC1CN2C(=O)CCC1CCCN1C(=O)CC(C)(O)C=C C1(NC(CNC(C(C)C)=O)=O)C2CCCN(C(=O)OC(C)(C)C)C2C1(C)C.C1(N)CC1 Cc1ccc(O)c(C(N2CC(CNC(=O)Cc3cc(F)ccc3O)CC2C)=O)c1 N1(C(=O)CC23CCCC2C3)CC2(CCN2C(c2csc(Br)c2)=O)C1 c1(C(=O)Nc2cc([N+](=O)[O-])ccn2)cc2c(c([N+](=O)[O-])c1)OCO2 CCC(CCCC(=O)N1CCCC1C1(C)CC1)NC(=O)CCSCC1CC1 c1(C(N2C(CC)CN(C(=O)CC3CC(OC)C3)CC2)=O)cc(C)cc(C)c1N c1(NC(N2CC3CC3(CO)C2)=O)nc(-c2ccccc2)nc2ccccc12 c1(CC)conc1C(=O)NC(Cc1ccccc1)CCNC(=O)Cc1cnns1 C#Cc1cnn(CC(=O)NC(CNC(=O)C=Cc2csc(C)n2)C2CC2)c1 C1(C(=O)NC(c2ccc(C(=O)NCC3CN(C(N)=O)C3)s2)C)C2CC2C2CC12 c1(C(=O)NCC2(NC(CC(=C)Br)=O)CCOC2)cc(N)c(F)cc1F N1(C(CCC2(C)CCO2)=O)CC(NC(=O)C(F)(F)NC(=O)C(F)(F)F)CC(F)C1 c1(C(=O)NC(C)CCCNC(C2CCCSS2)=O)ccc(-n2ccnc2)cc1 CCC(CNC(C1CCCCC1OC)=O)(CC)NC(c1ccc(OC)nc1)=O C(=O)(CC(=O)NC(C1CCOC1)CNC(C1CCCN1c1cnccn1)=O)OC c1(OC)cc(C(F)F)c(C(N2CC3CC3(CNC(C3(C)CCC3C)=O)C2)=O)cn1 C1(C(N(OC)CC2CCCCC2)=O)CCCCN(C(C2CC(C)C2)=O)C1 c1(OC)ccc(Cl)c(C(=O)NC2(C)CC(N(C3CCNCC3)C)C2)c1Cl N1(C(C(c2ccc(C)cc2)C)=O)CC2(C(N3CCOCC4(CC4)C3)=O)CCC1CC2 C1(CC)CN(C(C2CC=C(C)CC2)=O)CCN1C(c1cncc(OC)c1N)=O C(=O)(C1=C(C)CCC1)N1CCC(c2ccccc2)(NC(C=CC(CC)C)=O)C1 Cc1ccc(S(=O)(=O)N2CCN(C(c3c(C)cccc3Cl)=O)CC2CO)c(C)c1 CC(CN1CCOCC1)C(=O)NCC1CC(NC(C2CC=CCO2)=O)C1 C1(C(=O)NC23CC(C2)N(C(=O)CC2=CCOCC2)C3)CCc2[nH]nc(O)c2C1 c1(NC2C(NC(CC(CN(C)C)O)=O)CS(=O)(=O)C2)ncc(Br)cc1C#N CCC(CC)CC(=O)NC(C)(CNC(=O)C=Cc1cccn1C)CC N1(C(C(C2CCC(=O)N2)C)=O)CCC2C(NC(C3CC(C4CC4)C3)=O)C2C1 N1(C(C2CC(=C)C2)=O)CC(CNC(=O)Cn2cc(C(F)(F)F)cn2)(OC)C1 C=CCC(CC)C(=O)NC(CO)C(=O)NCC(O)CO C(=O)(CCCC(=O)N1CCN(C(=O)Cc2ccc(C)c(Cl)c2)C2CC12)NCCC N1(C(C2CCCSCC2)=O)CC2CN(C(=O)C(c3cc(F)cc(F)c3)O)CC2C1 C1(C(=O)NC(CC2CN(C(c3cnn(CC)n3)=O)C2)C)CCC(C)=C(C)C1 c1(OC)cc(C2(CNC(=O)C(C)O)CCC2)ccc1Br N1(C(c2c(C)cc(C)s2)=O)CCCC2(NC(c3cc4cc(Cl)sc4[nH]3)=O)CC2C1 C1(C)(CNC(c2cc(CCCC)c(NC)cc2)=O)CN(C(=O)CSC)C(C)(C)C1 C1(CNC(c2c(C)ocn2)=O)CC2COCC2N1C(=O)CC(C)C(F)(F)F C1(NC(C=CC=CCC)=O)CCCC2CN(C(c3ccc4cncn4c3)=O)CC12 c1(NC(C2CCN(C(c3c(C)cc(F)c(F)c3)=O)C2)=O)ncc(I)cc1[N+](=O)[O-] C1(C(=O)NC2CCCN(C(CCNC(C)=O)=O)CC2)CCc2nnc(O)cc2C1 C1(C)(CNC(C(CO)N(C)C)=O)CCC(NC(c2cc(F)n[nH]2)=O)C1 Cc1nc2cc(Cl)c(NC(C3CC(O)CN3C(=O)CO)=O)cc2s1 N1(C(c2cccc(C(C)C#N)c2)=O)CC2C(C(=O)O)(C1)CS2(=O)=O C1(C(=O)NCC2CC(CNc3cccs3)C2)CCCN1C(C1CC1(F)Br)=O c1(C(=O)NC2C(C)N(C(c3ccsn3)=O)CCC2)[nH]c2ccccc2c1Cl C12(C(=O)NC3CC(CNC(c4ncc(F)cn4)=O)C3)CCCCC1C2(F)F c1(CC)[nH]nc(C(=O)NCc2nc(CNC(c3cscc3OC)=O)cs2)c1Cl N1(C(C2CC(C)OCC2)=O)CC(C2CCCN(C(C3CCCC34CC4)=O)C2)C1 C1(NC(=O)CCc2ncc[nH]2)CCC(CNC(C2CC(F)(F)C2)=O)CC1 c1(C(=O)NOCC(c2n(CC=C)nnn2)CC2CC2)cccc(Cl)c1 n1(CCc2ccccc2)cc(COCC(N2CC(CN3CC4CC4C3)C2)=O)nn1 C1(CNC(c2cc(C(=O)OC)no2)=O)CCCCN(C(=O)CC2=CCCC2)CC1 CCC(CC(F)(F)F)NC(C1(CC)CCCN1C(=O)CCc1ccco1)=O C1(C(=O)NCCC2(OC)CN(C(=O)C(C)C)C2)CCS(=O)(=O)N1 CC1CC(C(=O)NC23CC(C2)N(C(C2CCCOC2C)=O)C3)CC(C)C1 CCC(C)C(C(=O)NCC1CNC(=O)O1)N(C(=O)C(C)COC)C c1(OC)noc(C)c1C(=O)NC(C1CCCC1)CNC(=O)C(c1nc(C)cs1)C C1(OC)CC(CNC(c2ncccc2C)=O)N(C(=O)C(N2C(=O)CCC2=O)C)C1 c1(CC(=O)N(CC(CC)NC(=O)CC2CNC(=O)C2)C)c(C)cccc1C C(=O)(C1=NOC(C)(C)C1)NC1CN(C(c2n(CCOC)ncc2)=O)CC1(C)C N1(C(c2ccc(SCC)nc2)=O)CCC(C)(C)C(NC(C2COC(C)C2)=O)C1 C1(CNC(c2ccc(Cl)cc2)=O)CN(C(c2snc(O)c2Cl)=O)C2CC12 C1(C(=O)NC2C(CNC(C(C(=O)OC)(C)F)=O)CCC2)CC12CCS(=O)(=O)CC2 c1(NC(COCC)=O)ccc2c(c1)CN(Cc1cccc(C)c1C)CC2 c1(C(N2CC(O)CC2CO)=O)cc2c(-c3ccc(O)c(F)c3)cccc2s1 N1(C(C2C(NC(c3c(Br)cnc(C)n3)=O)CCCC2)=O)CCC2(CCCO2)CC1 CCCC(CCCNC(c1ccc(Cl)cn1)=O)Nc1ncnc(Cl)c1C c1(C(N2CCC(NC(C(CC)=O)=O)C(C)(C)C2)=O)ccc2sccc2c1O C(=O)(C1CCCn2c(C)cnc21)NC1(CCNC(c2cncc(C#C)c2)=O)CC1 C(=O)(CN=c1[nH]c2c(c(=NC3CCNCC3OC)[nH]1)CSC2)N1CCC(OCC)C1 O=C1CC2CC(NC(=NCc3cc[nH]n3)NC(C3CC3)C3CC3)C1C2 C(=O)(CCC(=O)NCCNC(C1CCCCS1)=O)Nc1nnc(CC)s1 CC1CN(C(=O)CCc2cccnc2Cl)CC1NC(=O)C(C)c1ccsc1 C1(C(N(CCCC)CCO)=O)CN(C(c2snnc2C)=O)CCC1O N1(C(=O)COCC(F)F)CC2(CNC(C3CC34CC4)=O)CCC1CC2 C1(C(C)NC(C2(C3CCCO3)CCC2)=O)CCCN1C(=O)CNS(=O)(=O)C1CC1 N1(C(c2cnc(C)[nH]2)=O)CCC(C2CC2)(CNC(c2ccc(O)nc2)=O)C1 CCCC(C(=O)N1CC2=C(C1)CN(C(c1nocc1Br)=O)C2)C(C)C C1(N(C(c2cn(CC=C)nc2)=O)C)CN(C(c2occc2C2CC2)=O)CC12CC2 N1(C(CC(C(=O)OCC)(C)C)=O)CC2COCC(C1)C2NC(=O)C(C)CC(N)=O C(=O)(C(O)C(F)(F)F)N1CCN(C(C(C)Oc2cccc(Cl)c2)=O)CC1 CCC(CC(=O)NCC1CC(F)(CNC(C2CCCC2)=O)C1)Nc1nnn(C)n1 c1(C(=O)NC2C(CNC(C3N(C)CCC3)=O)C2)ccc(-c2ccccc2)c(F)c1 c1(C(=O)NCC2N(C(C(C=CCCC)O)=O)CCOC2)[nH]nc2ncccc12 C1(CNC(C(CC=CC)C)=O)CN(C(c2cnn(CCC)c2)=O)CCCO1 c1(C(=O)NCC(C)N(C)C(c2cc(Br)no2)=O)cccc(F)c1C#N C12(C(=O)NCC3CCC(NC(C4C(CC)OCC4)=O)CC3)CC(C1)S(=O)(=O)C2 C(CC(C)(C)C)(C(=O)N1CCC(F)(C(=O)NC2CC3CCC2O3)C1)OC C(=O)(C1CCCc2nncn21)N1CCN(CCn2cc(C(CC)O)nn2)CC1 N1(C(Cc2n[nH]c(=NC)s2)=O)CCCN(C(=O)C(C23CCCN2CCC3)OC)CC1 C1(CNC(C(CC)N(C)C)=O)CCCCC1CNC(=O)CCCN1CCCCC1 C1(NC(COCCCOC)=O)CC(O)CN(C(=O)CN2CCCNC2=O)C1 c1(C(=O)NCC2OCCN(C(CC(CC)O)=O)C2)cnn2ncccc12 C1(CC(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)CCC(C)(C)O1 c1(C(=O)NCC2CN(C(C3(CC)CCCC3)=O)C2)oc(C)nc1COC c1(CCC)ncc(NC2(c3nnnn3CC3CCOC3)CC2)cn1 C1(C(=O)NCC(CNC(=O)C(c2cccs2)SC)OC)CC2CCC1CC2 C#CCC(C)(C)C(=O)N1CC(C(N)=O)(CNC(C2CCCCN2C)=O)C1 C(c1cc(Cl)ccc1Cl)=CC(N1C(CNC(c2n[nH]c3c2COC3)=O)CCC1)=O C(CC(C)C)(C(=O)NCC1CN(C(c2cc(C#N)[nH]c2C)=O)C1)NC(C)=O C(=O)(C(=O)CCCCC)NC(CC(=O)NCCCC(=C)Cl)CCC c12ccc(cc1OC)CNC2=O.C1(C2CC2)(CC)CCCO1 C1(NC(c2cc(CCC)[nH]n2)=O)CCCCN(CCCC2CCOC2)C1 CC1CCCC=C1C(=O)NCC(CC(=O)NCCN(C)C)C1CCC1 N1(C(c2n(CC)ncc2)=O)CC(NC(=O)CCCN(C)C)CCC(O)C1 c1(C(=O)NC(CNC(C(CC)(C)CO)=O)C)[nH]c(C)c(S(N)(=O)=O)c1C c1(NC(N2CCC(CCCc3ccc(Cl)cc3)C2)=O)cccc(C(F)(F)F)n1 C1(CNC(C(C(CC)(C)C)O)=O)CN(C(c2sc(C)nc2C)=O)CCC12CCC2 Cc1ccc(CN=C(NC2CCCSC2)N(C)Cc2ncnn2C)cc1F N1(C(C2C(=C)C2)=O)CCC(F)C(NC(=O)CCc2nc(C(C)(C)C)no2)C1 C1(CNC(CC2(C)CC2)=O)(NC(c2ccc(C(F)F)nc2O)=O)CCCCCC1 c1(CC(=O)N(C2(CC(=O)NC(CC=CC)CO)CC2)C)ccc(C)nc1 c1(COCC(=O)NC(C)(C)CCNC(=O)CC2(C)CC2F)ccc(F)cc1 C(CCC(C(=O)NCCCSC(F)F)NC(=O)Cn1cnnn1)OC n1(CCC)nc(C)c(NC(=O)C(=O)NCC(c2cc(F)ccc2F)O)c1C c1(CCCC(=O)NCCN(CCOCCO)C(C2CC3CC3C2)=O)ccc(F)cc1 c1(CN=C(NC2CCC(C(N)=O)C2)NCCF)cnc2ccccc2n1 c1(CC(=O)NCC(C(C)C)NC(c2c(CC)nco2)=O)cnccc1C C1(CC)CN(C(c2conc2CNC(=O)C(C)n2cccc2)=O)CCN1C C1(NC(CC=CC=C)=O)CCC(C)(CNC(=O)Cc2ccc(Cl)s2)C1 CCC(C)CC(C(=O)N(C)CCC1CCCC1)NC(=O)CCOC1CC1 C12(NC(c3cc(C(C)(C)C)on3)=O)CCCC1N(C(=O)CS(N)(=O)=O)CCC2 Cc1c(F)ccc(C(N2CC3CC3(NC(=O)CSCC(F)(F)F)C2)=O)c1Cl CC1(CNC(C2(F)CCCC2)=O)CC(NC(=O)CSCC2CCCO2)C1 c1(C(N2CC3CN(c4c(C)ccc(=N)[nH]4)CC3C2)=O)cccc([N+](=O)[O-])c1Cl c1(NC(C2C(C)C2)=O)ccc(NC(c2ccc(O)cc2F)=O)cc1F C#CC1(C(=O)NCCc2cnc(C)o2)CN(C(=O)C(c2ccn(C)c2)C)C1 C(=O)(C(F)(F)C(F)(F)C(F)F)NC1CCC(CNC(=O)C2=C(Cl)CCC2)C1 O=C(CCCC(F)(F)F)NCC1CC1CC(N1CC2CCCC12)=O C1(C(=O)NC2CC(NC(c3cnc(C(C)(C)C)[nH]3)=O)C2)CCc2cncn2C1 c1(OC)cc(C)ccc1C(N1CCC(NC(c2cnoc2C)=O)C(C)C1)=O N1(C(CCC)=O)CC=CC1CNC(=O)C(C)(Cl)Cl C1(CC)CN(C(=O)CC2(C(F)(F)F)CC2)CCN1C(C1CCC1)=O C1(COC)(NC(=O)CC2CC2)CCN(C(C)=O)C1 N1(C(Cn2cc(C(C)=O)nn2)=O)CC2(CCC2NC(=O)C(C2CCCC2)OC)C1 N1(C(CCC#C)=O)CCCC(O)(CNC(=O)C(CC)NC(=O)CC=C)C1 c1(C(N2CCN(C(C3CCOC3)=O)C(CCO)C2)=O)cc(O)cc(Br)c1 C(CN=c1[nH]c2c(c(=NCC3CCOC3C(C)(C)C)[nH]1)SCC2)N(S(C)(=O)=O)C c1(NC(C2(C(=O)NOCC(F)(F)F)CCSC2)=O)cccc(CO)n1 C(=O)(C(CCN(C)C)NC(=O)CCc1ccncc1)NC(C)Cn1ccnc1 N1(C(c2c(OC)csc2)=O)C2CCC1C(CO)N(C(C1CCCN1C=O)=O)C2 CC1(C)CC(CNC(=O)CC(F)(F)Cl)CN1C(=O)Cn1cccc1 C12(NC(C(c3ccnn3C(C)C)C)=O)CC(NCc3cn(C4CC4)cn3)(C1)C2 C(=O)(C1=CC2CCCCCC12)NCCN(CC)Cc1nc(C)sc1C Cc1ccc(N2CCC(NC(=O)NCCc3cnc(C)o3)C2)c(C)c1 C1(OCC)CN(C(c2cnn(C(C)(C)C)c2)=O)CC1CNC(=O)CS(C)(=O)=O N1(Cc2ccc(OC)s2)CCc2cccc(Cl)c2C1.N12CCC3(CC3C1=O)C2 O=C(CC(F)(F)C(F)F)N1CC2(C(=O)NCC3(CF)CC3)CC1CCO2 C1(CCCCNC(c2cc(CC)[nH]n2)=O)CCCN(C(=O)CC2CC3CC3C2)C1 c1(C2(NC(C(C(C)OC)O)=O)CC2)cccc(C)c1F c1(OC)ccc(C(=O)NCC2(F)CC(NC(C3(C#N)CCCOC3)=O)C2)c(Cl)c1 c1(NC(c2ccc3c(c2)OCCO3)COC)ncnc2cc(F)c(Br)cc12 Cc1ccc(CC(=O)NCCCCCNC(=O)CC(C)c2cccnc2)c(Cl)n1 C12(NC(=O)CCc3ccc(Cl)c(F)c3)CCCC1CN(C(c1ccoc1)=O)C2 O=S(=O)(c1cncc(Br)c1)N1CCC12CN(Cc1nccnc1Cl)C2 c1(C(=O)NCC(C)(C2CC2)NC(CCCCCC=C)=O)cn2cccc(Br)c2n1 c1(C(N2C(CNC(c3cn(C)c(=O)cn3)=O)CC2)=O)nccn2c(Br)cnc12 N1(C(C(N2C(CC)CCC2)=O)=O)CC2CCCC(C1)N2C(=O)C(C)C1(O)CCC1 c1(C(=O)NCC23C(CN(C(C(COC)(C)C)=O)C2)C3)c(C)ncnc1C C(=O)(C(O)CC[S+](C)C)NCC1N(C(COCC)=O)CC(OC)C1 Cc1c(C(=O)NCCC2CCCN(C(=O)CC(C)c3ccco3)C2)ncn1C C12(OC(c3[nH]nc(N(C)C)n3)=O)CCCC1N(C(=O)OC(C)(C)C)CC2 c1(C(N(C2CCC(NC(C(C)NC(COC)=O)=O)C2)C)=O)cnc(OC)nc1 n1(CC(=O)NC(CC)CNC(C23CC(CN2C2CC2)C3)=O)nc(C)c2cccnc12 C1(C(=O)Nc2cc(C)cc(C)c2)CC2CC1CN(C(=O)Cn1nc(C)cc1C)C2 c1(NC(C)=O)cccc2c1CCN(CC(N1CCOCC3(C1)CC3(F)F)=O)C2 c1(CC)ncncc1C(=O)NCC(C1CC1)NC(=O)Cn1ccnc1C C1(C(=O)NCCN(C)C(c2cnn(-c3ccc(Cl)cc3)n2)=O)CC(C2CCCC2)C1 Cn1cc(NC(c2nnnn2C2CC(F)(F)C2)c2ccco2)c(O)n1 C(=O)(C#CC1CCOC1)NC(CCC(=O)NCC1(OC)CCCCC1)(C)C N1(C(C2CCC(CC)O2)=O)CC2OCCN(C(=O)Cc3ncc(CC)[nH]3)C2C1 C1(NC(c2c(C)coc2)=O)CN(C(c2n[nH]cc2Cl)=O)C2CCCCC12 C(=O)(CC(Cc1ccccc1)CC)NCCCNC(C1N(C(C)=O)CC(O)C1)=O CC1CN(C(=O)Cc2ccn(C(F)F)n2)C(C)CN1C(=O)CSc1nnc(S)s1 N1(C(C2(NC(CC(C)OC)=O)CC(O)C2)=O)CCC(CC(C)O)CC1 c1(N2CCC(C(=O)OC)CC2)nc2ncn(C)c2c(=NCC2(C)CSC2)[nH]1 c1(C(CNC(C2CCN(C)CC2)CC)C)cc(F)cc(F)c1 c1(C(=O)NC2CCC(NC(=O)CCCF)CC2)c[nH]c2cccnc12 C12CCN(CC1)C2=O.O=C(O)CCOOC1CC1.C1CO1 n1(CCC(=O)NC2CC(C)N(CCc3cnccn3)CC2)cnc2ccccc12 C(c1nnc(C(C)C)o1)=CC(=O)N(C)CC1CN(C(C(CC)C)=O)C1 c1(CNC(C(=O)OC)C2CN(C(=O)OC(C)(C)C)C2)nc2n(c1Cl)CCCC2 C(=O)(C1c2ccccc2C2CC1C2)NCC1(CS(=O)(=O)CNC(C)=O)CCOC1 C1(N(C(C(C)n2cccn2)=O)Cc2cccn2C)CC12CCNCC2 Cc1cc(C#N)ccc1-c1cn(C(C)CNC(=O)CNC=O)nn1 O=CN1CCCC1C(=O)NC(C(=O)NCC(F)(F)CC1CC1)C1(O)CCC1 CCN=C(NCc1ccc(C(N)=O)o1)N1CCN(C2CCNC(=O)CC2)CC1 C1(NC(C(CC(C)C)=O)=O)CCCC2CN(C(=O)CCC3CC3(Cl)Cl)CC12 c1(OC)ccc2ccccc2c1CN1CCCC1C(=O)Nc1ccc(C)nc1C N1(C(C=C(CC)C)=O)CCOCC1CN(C(=O)CN(C)Cc1ccc(Cl)s1)C c1(C(N2C(C)CC(CC(=O)NCc3cc(N)ccn3)C2)=O)cnc2[nH]cnc2c1 C(=O)(C#CC1(C)CCCO1)N(C1CCN(C(c2nncs2)=O)CC1)CC c1(C(N2CC(c3cn(CC(COC)O)nn3)OCC2)=O)cccc(F)c1Br C1(NC(c2cn(C(C)C)nn2)=O)CCN(C)C12CCCN(C(c1cc[nH]n1)=O)C2 C(=O)(C(O)CC(F)(F)F)N1CCN(C)CC1C(=O)NCCSCCCO CC(C)CC(C)(CN)C(=O)N1CCCC1Cc1cccc(Br)c1 C(=O)(CCCCC#N)N1CCN(C(CNC(C2OCCC(C)C2)=O)C)CC1 c1(N2CCC=C(C(=O)NC3CCCC(F)C3)C2)ncc2[nH]cc(I)c2n1 c1(C(N(C2CCN(C(=O)CC3CC4CC4C3)C2)C)=O)nn(C(F)F)cc1Cl C=CCC(CNC(=O)Cn1cc(-c2ncccc2C)nn1)C(=O)N1CCCCCC1 C12CCC(O)CN(C1)C(=O)N2.C1(C)(C(=O)NCc2onc(CC)n2)CCSCC1 c1(CC)c(OC)ccc(C(N2CCCCC2CNC(C2CCO2)=O)=O)c1OC CCC(CC(=O)N1CCCC1(C)CCC(=O)NC1CCOCC1)OC C1(CCNC(CNC(N)=O)=O)CCCCN1C(=O)Cn1ncccc1=O C(=O)(CCCC(=O)N1CC(CNC(=O)C=CC(C)(C)C)C2CC12)N(C)C C1(NC(CCC(N)=O)=O)CC2CC(NC(c3cnc(O)c(Br)c3)=O)C2C1 CCCCCCCC(=O)N1CCCC(C(=O)NC(C)CCC2CC2)C1C Cc1cc(F)cc(C)c1CN1CCC(NC(c2ccnnc2O)=O)C1 C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CN(C(=O)Cc2nocc2C2CC2)C2CC12 C(=O)(CC(C(=O)N1CC(NCc2cc(=O)cc[nH]2)CC(C)C1)c1ccccc1)OC C1(CNC(C2(SC)CC2)=O)CN(C(=O)CNC(=O)C(C)(C)C)CCC12CCOCC2 c1(C(=O)NCCC(C)NC(C(C2CCCC2)OCC)=O)c[nH]c(C(F)(F)F)c1 c1(C(N2C(CNC(CCCCC=CC)=O)CC2)=O)cnc(N)c([N+](=O)[O-])c1 CC1CCCN(C(C2CN(C(=O)C(N)=O)CC2C)=O)C1CO c1(OC)ccc(OCCC(N2CCC(NC(C3CC(=O)N(O)C3)=O)CC2)=O)cc1 C1(CNC(=O)CCn2cccn2)COCCN1C(C1CCC1CF)=O O=S1(=O)CCC(O)(CNC(=NCCc2cnco2)NCC(=O)NCC(F)F)C1 CCCC(C(O)C(=O)Nc1ccc(C)nc1C)NC(c1cc(Cl)cn1C)=O C(C(C(=O)N1CCC(C(C)C(=O)NC)C1)NC(=O)CCCC1CCC1)OCC C=C(C)CC(C(=O)N1CCOC(CC(=O)NC(c2nccn2CC)C)C1)OC c1(OC(CNc2c(C)n[nH]c2)(F)F)ccccc1C N1(C(C(COC)C)=O)CCCC12CCC(NC(=O)Cc1nnc(S)n1C)CC2 C(=O)(CC1OB(O)c2ccccc21)NCC(C)CNC(c1ncc(Cl)cc1Cl)=O C(=O)(CCC(C)(C)C(=O)NC1CN(C(c2ccco2)=O)CC1OC)OC C1(C(C(=O)NC(CCNC(C2CC(C(C)C)C2)=O)C)O)CC(F)(F)C1 CC(C)CC(=O)N(CCC(=O)NC(C)(CCC(C(=O)N)O)c1nn[nH]n1)C1CC1.N(C)C C(=O)(C1(C)CCOc2ccccc21)NCC(C)(C(=O)NC1CN(C(C)=O)C1)OC c1(CCN=C(NC(CC)C)NCC2CN(C)CCO2)nc2ccc(Cl)cc2[nH]1 c1(SCCN2CCNC(=O)C3C(C3)C2=O)ccccc1CC.C(=O)OC C1(NC(C(=O)NC(c2ccc(Br)cc2)C#C)=O)CC2(CCC2)C1O C1(NC(C2OCC(C)C2)=O)CCCC2CN(C(c3nnn(C(C)(C)C)n3)=O)CC12 N1(C(c2cn(C)nn2)=O)CCCCC(CCC(=O)NCc2nn(C)c(=O)n2C)C1 CCS(=O)(=O)c1ccc(CNC(C2(C3CC3)CCCNC2)=O)s1 Cc1cc(NC(C2CC3CC3N2C(=O)CCSC2CCCC2)=O)cc(Cl)c1 C1(CNC(C=CCN(CC)CC)=O)CCCCN(C(c2nc(C)no2)=O)C1 N1(C(C(=O)NC2C(C)CC(C)(C)CC2)=O)CCc2ncccc2C1 C1(C(F)F)(CNC(Cc2ncc(C)[nH]2)=O)CCN(C(=O)C(C)OC2CCCC2)C1 C1(C(=O)NC2CCC(NC(c3cncc(C)c3)=O)C2)CN2CCC1(C)CC2 C12(NC(c3nc(CCC)oc3)=O)CC(CNC(=O)CN(C)C)(C1)OC2(C)C c1(C(=O)N(CC(C2CCOCC2)(C)C)C2CC2)cc(C(F)(F)F)n[nH]1 C1(CNC(c2ccc(CC)[nH]2)=O)CC(NC(c2ccc(N)cn2)=O)C(O)C1 c1(N2CCC(C)C2CNC(c2ccc3nonc3c2)=O)ncnn2c(Br)ccc12 C=C(C)C(CC(=O)N1CC(NC(c2cc(Cl)ccc2CC)=O)CC(C)C1)OCC C(=O)(C1=CCOCC1)NC(CCCNC(C(C)Sc1ccccn1)=O)(C)C C(=O)(C1c2ccccc2OCC1(C)C)NCCNC(C(CC=C)(C)C)=O N1(C(C2C=C(C)CS2)=O)CCC2(C=C(C(=O)N3CCOC(CC(C)C)C3)C2)C1 c1(C(=O)OC)cc(C(=O)NCC(C)(O)CNC(=O)Cc2cccnc2C)c(C)o1 c1(N2C3CC(CNC(c4c(CC)csc4)=O)C2CC3)cc(C)nc(S(C)(=O)=O)n1 CC(C)CCC(=O)NCC(=O)NC1CCC(N(C)C(C2C3CC3C3CC23)=O)CC1 c1(C(=O)NC2C(NC(C(CC#C)C)=O)C2)cnc(CC2CC2)nc1O C1(COC)(NC(=O)CC2CCCCC2C)CCN(C(=O)CCc2cccnc2)C1 N1(C(C2(C)CC2C(F)(F)F)=O)CCC2CCC(C1)N2C(c1ccc2oncc2c1)=O O=C(CCCF)NC1CCC1C(ONC(C1(NC(=O)C2CC2)CSC1)=O)=O C1(NC(=O)Cc2ccncc2Cl)CC2CCC1CC2NC(C1(O)CCCC1)=O C(CC1=CCN(C(=O)Cc2cnc[nH]2)CC1)NC(C(=Cc1ccccc1)OC)=O C(=O)(CC(C)C(C)C)N1C(CNC(C(COC)COC)=O)CC1 c1(C(N(C2CC3CCC(C2)N3C(c2cn[nH]c2)=O)C)=O)cccc2c1CCCN2 c1(C(N(C2CC(NC(=O)CCP(C)(C)=O)C2)C)=O)csc(S(C)(=O)=O)c1 N1(C(c2n(CC)c(O)nc2)=O)CC(NC(c2nc(C3CC3)oc2C)=O)CCC1C Cc1cc(C(N2CC=CC(NC(C3CC3F)=O)C2)=O)n(CC(F)F)n1 C(CC(CC)C(=O)NCC1CCCCN(C(=O)C(=O)NCC)C1)=CC N1(C(CNC=O)=O)CC2CCCC(C1)N(C(C1COCCN1CC(F)(F)F)=O)C2 C1(N(C)C)CS(=O)(=O)C12CCC2.Cc1nn(C2CCCCCCN(C)C2=O)cc1Cl C(=O)(CC1OCc2ccccc21)OC(C)CC1=CCCCC1 c1(NC(C2N(c3ncc(C(=O)OC)cn3)CC(C)C2)=O)cc(Cl)cc([N+](=O)[O-])c1O c1(CC(N2CCC(CCN(C(=O)CO)C)CC2)=O)cccc2ccncc12 C1(O)(CCNC(c2cc[nH]n2)=O)CCN(C(C2CCC2c2nc[nH]n2)=O)CC1 CN(S(=O)(=O)N1CCN(C2CCCCC2O)CC1)C1CCCC1 c1(C(=O)NCCN(CCOC)C(c2cnn(C3CCC3)c2)=O)ncsc1C C1(N(C(c2cc(C#C)c(OC)cc2)C(=O)NCC=C)C)CCN(S(N)(=O)=O)CC1 C1(C)(CC)CC(NC(=O)C=Cc2ccncc2)CN1C(=O)C#CC1CC1 c1(C(=O)NCCCCNC(C2(C)CCCN2)=O)cccc(F)c1 c1(CC(=O)OC)nc2ccc(NC(=O)NC3CC3(c3ccccc3)C)cc2s1 C(C(C)CC(=O)NCC(CC(=O)N1CCCCCC1)C1CCC1)OC C(C)(C(=O)NC1CCSC1)NC(CSCC)=O N1(C(C(C)SC)=O)CCCCC(NC(=O)CCN2CCC2)C1 C1(NC(c2c(C)oc(-c3ccc(C(F)(F)F)cc3)n2)=O)CC12CCC(C)(C)CC2 c1(OC)cnc(Cl)c(C(N2CC=CC(NC(C3(OC)CCC3)=O)C2)=O)c1 c1(C(=O)NCCC(C)NC(=O)CC2CCCCCC2)cccc(Cl)c1 c1(OC)cn(CC(=O)NC2CN(C(c3cc(F)n[nH]3)=O)CC2OC)c(C)cc1=O N1(C(C(=O)NCC(F)C2CC2)=O)C2CCC1CC(=O)C2 C(=O)(CCC(=O)NCc1cccnc1C(N1CCN(C2CCC2)CC1)=O)NCC N1(C(c2c(C)nsc2C)=O)CCC2(CC1)CC2NC(c1ccc2c[nH]nc2n1)=O c1(C(=O)NCCC(C)NC(C2C(=C)C2)=O)cnc2ccnn2c1N c1(C(C(N2CC(O)(CCNC(CCc3n(C)ccn3)=O)C2)=O)O)cccc(F)c1 c12ccc(cc1)SCC(C)(C)CN(C)C(=O)CO2.N1(C(CCC)=O)CCCC1CC C(=O)(C(=O)N=S(C)(C)=O)NCC(CN(C(c1cc(COC)sc1)=O)C)C C12(CNC(c3scc(CNC(CCC(=O)NC)=O)c3)=O)CCC(CC1)CC2 C=CCC(C)(C)CC(=O)NCC1CC(C)CN(C(c2cccc(C)c2C#N)=O)C1 c1(C=O)cc2cccnn2n1.C1(CN2CC(n3cc(CC)nn3)C2)CC2CCCCC12 c1(-c2ccc(C(C)O)cc2)ccc2ccc(C(N3CC4COCC4C3)=O)nc2c1 C12(NC(c3ncsc3CC)=O)CCC(NC(c3ccc(Br)nc3OC)=O)(CC1)C2 CC(CC(=O)NCC1CC(NC(=O)Cc2ccc(Br)cn2)C1)C(F)F c1(-c2ccc(COC(F)F)[nH]2)nc(-c2cccc(Cl)c2)nn1-c1cccc(Cl)c1 c1(C(N2CCCC(NC(c3n(CCC)ccc3)=O)CC2)=O)cc(Cl)c(F)cc1O C(=O)(C(C)CC(=O)NC1C2CCCCCC12)N1CC(OC)C(C(=O)OC)C1 N1(C(COCCOC)=O)CC(CNC(C2(C(N)=O)CC2)=O)C(C)(C)C1 N1(C(c2c(C(=O)OC)con2)=O)CCN(C(C23CCC2CC3)=O)C(C)C1C CCC(CC(=O)N1CCN(C(=O)CCOC2CC2)C(C)C1)CC(F)(F)F CC(C)CCC(F)C(=O)NCc1cncc(C(N2CCC(CO)C2(C)C)=O)c1 C1(C(C(=O)NCCC)N(C2CCN(S(C)(=O)=O)C2)C)CCC(C)(C)CC1 C1(NC(C(n2ncc(C)c2)C)=O)(CO)CCCN(C(c2ccnc(CO)c2)=O)C1 N1(C(C2C(C#N)C2)=O)CCc2c(CNC(C3CC4CCC3C4)=O)cccc2C1 c1(C(N2CCCC(O)(CN(C(C(C)SC)=O)C)C2)=O)cnc2[nH]ncc2c1 C1(NC(c2c(C)nccc2)=O)CC2CC1N(C(=O)COc1ccc(Cl)cn1)C2 C#CC1(O)CC(C(N2CCC(O)(CN(C)C(c3c[nH]nc3Cl)=O)C2)=O)C1 C12(NC(CCC(C)(C)OC)=O)CCCC1CN(C(c1ccncc1Cl)=O)C2 N1(c2nccc(=NCc3cnc(C#N)s3)[nH]2)CCSC2(CCOCC2)C1 c1(CSC)cn(CC(C)(C)CNC(C2(c3ccccc3)CC(O)C2)=O)nn1 c1(N(C2(COC)CCC2)C)cc(Br)ccc1S(=O)(=O)NCC1CCC(OC)C1 c1(CC)nc(Cl)c(C)c(=NC(C)C2CCN(C(=O)C#CC3CCCCO3)CC2)[nH]1 N1(C(c2cnc(C)s2)=O)CCC2CC2(C(=O)N(C)CCOC)CC1 C1(C(N2CC(CN(C(C(COC)N(C)C)=O)C)C2)=O)COCC1(C)C CS(=O)(=O)c1ccc(C(N2CCN(C(c3cnn(CCO)c3)=O)C3CC23)=O)cc1 C1(NC(CN(C)CC)=O)Cc2ccccc2C1NC(C1(C)CCOC1)=O N1(C(C2(C(C)(F)F)CC2)=O)CC2ON=C(CNC(c3csc(F)c3)=O)C2C1 CCCCC(O)C(C)C(=O)N1CCC(NC(c2ccc(OC)nc2F)=O)C1C C1(N(C(=O)COCc2cccc(CC)c2)CC#C)CCN(C(C2CCC2)=O)CC1 C1(Cl)(C(N2C(C)C=C(CNC(C3OCC4CCCC34)=O)CC2)=O)CC2CCC1O2 CC1CC=C(C(=O)N2CCN(CCCNC(C3CCCNS3(=O)=O)=O)CC2)CC1 CCC(CC(C)C)C(=O)N1CCCCC1O[Si](C)(C)C(C)(C)C c1(CN(C(=O)CC2CC(CC(N3CCOC(CC)C3)=O)C2)C)ccc(F)c(F)c1 c1(C(C(=O)NC2C(NC(c3ccncc3)=O)CC2)O)ccccc1C(F)(F)F C1(NC(c2n(C)nc(C)c2F)=O)CCSC12CN(C(c1ns[nH]c1=O)=O)C2 N1(CCOC)CCN(C(=O)C(C)(C)C2CCCN2C(=O)CCC2CC2(C)C)CC1 C1(CNC(Cc2c(C)noc2C)=O)CC12CCN(C(=O)CCC1CC1(C)C)CC2 c1(C(c2nnnn2CCC2CC2)NC(c2ccc(C)cc2)CC)ccncc1F N1(C)CCOCC1C.c1(CC)nnsc1CNC(CC)CCn1cc(CCOC)nn1 C1(C)(C(N2CCC(N(C)CC)CC2)=O)CN(C(C2CCCCN2C)=O)C(C)(C)C1 C1(CNC(Cc2c(C)cccn2)=O)CCCC2CN(C(c3cc(Cl)no3)=O)CC12 c1(C(=O)NC2C(CNC(CN(S(CC)(=O)=O)C)=O)CC2)cn(C)ccc1=O CCC(C)CC(C(=O)N1CCCC1CF)NC(=O)CC12CCC(CC1)C2 N1(C(=O)OC2CCNC2=O)CCN(CC(O)COc2ccccc2)CC1 N1(C(C)=O)CCOC(C(=O)NCCCC(C)NC(C2CCN(C)CC2)=O)C1 C1(C2CCOCC2)(C(N2CC(COC)C(NC(C(C(CC)C)OC)=O)C2)=O)CC1 CCCCC(CN1CCOCC(C=O)C1)CC.S(C(F)(F)F)CCO C1(C(N2CC(NC(C(CC)N3CCCC3=O)=O)C(C)C2)=O)CN2CCN1C(C)C2 S(=O)(=O)(c1csc(C(=O)NCC2CCN(C(=O)CCc3cnc(C)o3)C2)c1)NC N1(C(c2nn(C)c3c2CCC3)=O)CC2CCC(C1)N2C(C1CCOC1=O)=O C(=O)(CCCCCCCCC1CCN1)N1CCN(c2cn(C(C)(C)C)nc2)CC1 C1(NC(c2n(CC)nc(C3CC3)c2)=O)CN(C(c2cnc(O)s2)=O)CCC1F c1(OC)cc(CC(=O)NC(C)C(C)NC(c2cnc(SC)s2)=O)ccc1C O=C1NCC2(CCCCC2)C(=O)N1Cc1cnc(C(F)(F)F)nc1 C(=O)(C1=CCCCO1)N1CCC(CCCCNC(C(C)CC2CCC2)=O)CC1 C(=O)(CC(C)C(C)(C)NC(=O)C(O)CN1CCCC1)NC(CC)C(=O)NC c1(C(N2CCN(C(c3c(C)con3)=O)C(CF)C2)=O)ccc2c(c1)CCO2 c1(C(N2CC3C(Nc4c5ncn(C)c5ncn4)C3C2)=O)cccc2ncccc12 C1(NC(CN(CC)CC)=O)CC2CSCC(C1)C2NC(=O)CC1CC1(C)C c1(CC)ccc(C(=O)NCC(CO)NC(c2ccc(SC3CC3)cc2)=O)nc1 C1(NC(CC)=O)CCN(C(=O)CCSC)C1.N12CC(C)(C1)CC2=O O=C1CC(NC(=O)C(N2CCCC(Cn3cccn3)C2)=O)CCN1 Cc1cc(C)cc(C=CC(=O)NCC(C)(C)CNC(C2CC2c2cccs2)=O)c1 C=CCC(CC=C)C(=O)NC1CCC(NC(c2ncc([N+](=O)[O-])n2C)=O)CC1 C(=O)(CCCCC(C)(C)OC)NCC1(C)CCC(NC(CCCOCC=C)=O)C1 CN1CCC(CC(=O)NC(C)(CO)C(=O)N(C)CC2COCCO2)C1=O C(=O)(CS(=O)(=O)N(C)C)NCC(CC)NC(C12CC(OC)C1C2)=O C1(CC(=O)NCC(c2ccccc2)OC)CN(C(c2cccs2)=O)CCO1 CN1CCOC(C(N2CC(O)(CNC(=O)CCCc3ccsc3)C2)=O)C1 N1(C(CN(C)C)=O)CCC2C(CCCN2C(c2cnc3nccn3c2)=O)C1 C1(NC(c2cc(C)n(C(C)C)c2)=O)CC(C)CN(C(=O)Cc2cc(Cl)n(C)n2)C1 c1(C(=O)NCC(C)N(C(=O)CCOCC(F)F)C)ncn(C)n1 C(=O)(C(C)(C)CC(=O)N1CCC(NC(C2CC(F)(F)C2(C)C)=O)C(C)C1)OC O=C1CCC(CC(=O)NCC(C2CCOC2)NC(=O)CNS(N)(=O)=O)N1 C12(NC(c3nc(COC)oc3)=O)CC(C1)N(C(c1ccc(Cl)cn1)=O)C2 c1(CC(=O)NCCC2(O)CN(C(=O)CN3CC4CC4C3)C2)cncc(F)c1 c1(OC)cc(C#N)ccc1C(N1CCC(F)(CNC(C2CC=CCO2)=O)C1)=O Cc1cc(C(N2CCC(O)(CNC(=O)COC3CCCOC3)C2)=O)cn1C(C)C C=C1CCN(C(=O)C(C)CC=CC)C(C(N2CC(CO)C(C)C2)=O)C1 CC(C)(C)C(CNC(C1CC1C1(C)CNC1)=O)C(=O)NOC1CCOCC1 N1(C(CC=C)=O)CCCC(N(C(=O)CCc2c(C)nn(C)c2C)C)CC1 Cc1cc2c(C(=O)NCC3CC3CNC(=O)Cc3ncc(C)s3)ccc(C)c2[nH]1 C(=O)(C1=CCCCCC1)NC12CCN(C(C3(CN(C)C)CC3)=O)CC1C2 C1(C(=O)NC2(C)CN(C(c3cc(CN4CCCCC4)on3)=O)C2)CCCOCC1 c1(C(=O)NC(C(C)NC(CC(CCC)O)=O)CO)c(C)ccc2c1CCCN2 N1(C(CS(CC)=O)=O)CC2(C1)CN(C(C1CC3(CSC3)C1)=O)CC2CO CCC(C)(C)C(O)C(=O)N(C1CN(C(c2cnc(C(C)(C)C)nc2C)=O)C1)C C1(CNC(CNC(=O)OC)=O)CCC1NC(=O)CCOC.C1CC1 c1(C(=O)NCCCCNC(C2CC(CC)C2)=O)c(F)cc(Cl)cc1Br C(c1cn(C)nn1)=CC1CC1.C1(=O)C(C)N(CCC)C(=O)N1CC#C c1(OC)ccc2c(c1)OC(CN1CCC(=O)N(Cc3cc(C)cc(C)n3)C1=O)C2 CC#CCCCC(=O)N1CCC(C(C)NC(=O)Cc2cccc(N(C)C)c2)C1 c1(OCCN(CC(=O)NC(c2ccccc2)C)CC)ccc(C)cc1 Cn1nc2c(c1O)CCN(c1nnc(CN3CCOC3=O)n1C)C2 c1(C(=O)O)cccc2c1CCC2NCc1c(Cl)cnc(F)c1Cl C12=CC(=NC(=O)NC1)NN2.CC1CC(C#N)CN1C(=O)OC(C)(C)C c1(NC(C2N(Cc3cc(C)c(F)nc3)CC=C2)=O)cc(Br)c(F)cc1F Cc1cc(C(N2CCCC2C2(NC(=O)Cc3nc(=N)[nH][nH]3)CC2)=O)cc(Br)c1 Cc1sc2ncc(C(=O)NCC(C)NC(c3c[nH]cc3C3CC3)=O)c(=O)n2c1C C(C(CN=c1cc(C)c(C#N)c[nH]1)C(F)(F)F)NC(C(CC)CC(F)F)=O O=C(C1CCCc2c(O)cccc21)NCCC1(O)CN(C(C2CCC2CF)=O)C1 N1(CC(CN2CCCC(CC#N)CC2)O)C(=O)NC2(CCCCC2)C1=O C(=O)(C(C)(C)C(=O)NC(C1CCCN(C(c2ccc(Cl)cc2)=O)C1)C)NC N1(C(c2n(C)c(Cl)nc2)=O)CCC(C(=O)NC2CC3OCCCC23)C12CC2 c1(C(N(C2CN(C(=O)COCCF)CC2F)C)=O)ccc(N)cc1F C(=O)(CCC(=O)N1CCC(CCNC(c2ccoc2I)=O)CC1)OC C1(F)(C(=O)NC(C)CCO)CCN(C(=O)Cc2sc(O)nc2O)CC1 CCS(=O)CC(=O)N1CC(CNC(c2ccc(C3(C)CCO3)cc2)=O)C1 c1(C(=O)NC(CNC(C2COC3(CCC3)C2)=O)CO)ccc2c(n1)CCC2 CC(C)(C)C(C(=O)NC(CNC(=O)CC(F)(F)Cl)C1CCC1)C1CCC1 CN1CCN(C(=O)C2=CCCSC2)CC1C(N1CCC2(CCO2)C1)=O C1(C(=O)NC2CCCCC2F)CC12CCN(C(=O)C=Cc1ccoc1)C2 c1(C(c2nnnn2C(C)C)N(C(C)C)C2CC2)conc1C1CC1 c1(OC)ccc(CC(=O)NC2CC(NCc3noc(C)n3)C2)c(OC)c1 C1(NC(c2cc(C(C)C)on2)=O)CCN(C(C2CC(C)(O)C2)=O)C1C1CC1 Cc1cn2c(C(=O)Nc3ccc4occc4c3)cnc2s1 C(=O)(C(F)(F)CCc1ccccc1)NC(CC(C)NC(c1cnc(OC)s1)=O)C CCC(CCCC(=O)NC1(c2nc[nH]n2)CC1)NC(C1CCO1)=O C1(CC=C)(NC(C23CCC2CC3)=O)CCN(C(c2cc(Cl)ccn2)=O)C1 c1(-c2scc(OC)c2)ccccc1C(=O)NCC1CCC(=O)N1C C1(CNC(c2coc(COC)n2)=O)CN(C(C23CC(C(=O)OC)(C2)C3)=O)CC1C C=CC(CCC)CC(=O)N(CC(F)C(=O)NCCCC)CC(=O)OC C(CC(=O)NCC(C1CCCC1)C)(C(F)F)NC(C(C(=O)OCC)OC)=O N1(C(C(C)C(F)F)=O)CCCC(O)(CN(C)C(C2(NC(N)=O)CCCC2)=O)C1 C(CCC(C)NC(N(C1CCOCC1)CC1CCCO1)=O)OCC c1(OCC)ccc(CC(=O)NCCN(C(=O)CCc2cnc(C)s2)C)cc1OC c1(C(=O)NCC2CCCCO2)c(NCCOC(F)(F)F)cccc1F c1(C(N2CC3(CC(NC(=O)COCC4CC4)C3)C2)=O)cc([N+](=O)[O-])cc(Cl)c1Cl c1(C(=O)NC23C(CN(C(C4(OC)CCC4)=O)C2)CCC3)ccn2c(O)nnc2c1 C(=O)(C(C)(C)CS(N)(=O)=O)NC(C)CNC(C12CCCCC1C2(F)F)=O Cc1cc(F)c(C(N2CCC(C)C2CNC(=O)C#CC2CCC2)=O)cc1Br C(=O)(CC(C(F)F)N1CCOCC1)NCC1CN(C(c2c(C)noc2C(F)F)=O)C1 N1(C(c2cn(CC)nc2)=O)CCC2(CC2)CC1C(N1CCN2CCC1CC2)=O c1(C(=O)NCC(C2(O)CCN(C(=O)CC(C)(C)O)C2)C)cc2n(n1)CCC2 c1(OC)cncc(C(=O)NC(C)(CSC)C(=O)NC2CCCCC2CO)c1 CCCC(F)C(=O)NN1CCC(C)CC1.c1(C(C)C)cnncc1CC(=O)O C=CC(C)(CCOC)C(=O)NC1CC2(CCC2)CN1c1ncccc1C(C)=O N1(C(C2(CC)CCCCO2)=O)CC(CN(C(=O)CCF)C)C2(CC2)C1 CN1CCOC(C(=O)NCCCN(C)C(c2cnc(-n3cccn3)cn2)=O)C1 C(=O)(CC1=CCN(C(=O)OC(C)(C)C)CC1)Oc1c(O)cc(C)c(Br)c1 C#CCCC(O)C(=O)NCCN1CCN(C(=O)CC2C(C)(C)C2(C)C)CC1 c1(C(C(=O)NC)N(C2CCN(CC3CCC3)C2)C)cccc(OC(F)(F)F)c1 CCC(CC)C(C(=O)N1CCC(O)C(C(=O)N(C)CCc2ccccc2)C1)OC C1(OC)(CNC(=O)C(C)CN(C)C)CCN(C(c2c(C)[nH][nH]c2=N)=O)C1 N1(C(CCC2C(C)C2)=O)C2CCC1C(CNC(c1ccccc1SCC#N)=O)C2 N1(C(CS(CC)=O)=O)CCC(CO)C(NC(=O)C2CC2)C1 C1(C(N2CCN(CCN(C)C)CC2)=O)CC2CC1CC2NC(=O)CC1CCCC1 C=CC1CCCC(NC(=O)CC2C(NC(c3ccsc3)=O)CC2O)C1 C1(C(N(C2CC2)CC2N(C(CN(C(C)=O)C)=O)CCC2)=O)CC(=O)N(C)C1 N1(C(C(CC)CC(C)C)=O)CCCC2(CCCCC2NC(=O)CC(C)(C)CC)C1 c1(CNC(N(CC(C)C)CC#C)=O)ccc2c(c1F)CCCC2 C1(C(N2CCC(C(C)(C)NC(c3cnccc3Cl)=O)C2)=O)Cc2nncn2C1 c1(C(c2ccc(C)cc2)N(CC(CSC)O)C)cc(Br)ccc1Br c1(N2C3(CNC(C(C)C4CCCO4)=O)CC(C2)C3)ncnc2c1c(Br)nn2C c1(C(N2CCC(C)C(NC(c3ccc(C)o3)=O)C2C)=O)ccc2c(c1)CCCS2 c1(C(N2CCC(C(CNC(C(NOC)=O)=O)C)CC2)=O)ccc(OC)cc1C C1(C(N(CC(C)CNC(c2ccnn2CCF)=O)C)=O)CCCNC1=O S(=O)(=O)(C(C)CCN)NC(c1c(-c2c(C(C)C)cccc2)cccn1)=O C1(C(=O)NCC2(NC(c3cc4scc(C)c4[nH]3)=O)CC2)C2Cc3ccc(Cl)cc3C12 C(=O)(CC(C)(C)C(=O)N(C)C)N1CCC(CCNC(C2CC(CCC)C2)=O)C1 Cc1cc(C)c(CNC(c2ncoc2C(F)F)c2nnnn2CCCF)cn1 C1(F)(CNC(C2C(C(=O)OC)C=C2)=O)CCN(C(=O)C(F)F)C1 C(N=c1cc(C)[nH]c(=NCC=CC(C)CC)[nH]1)c1cc(CC)no1 C1(CCC)(NC(=O)CC=Cc2ccccc2)CCCN(C(=O)CS(N)(=O)=O)C1 C1(NC(CCOCCC)=O)CCN(C(C23CC4CC2C3C4)=O)CCC1(F)F N1(C(C2CCN(S(CCCC)(=O)=O)CC2)=O)CCS(=O)C(C)C1 Cn1nccc1C=CC(N1CC2CC1C2NC(C1CCCO1)=O)=O CC(CCN=c1cc(C(F)F)nc[nH]1)NC(C1(C2CCCCC2)CC1)=O N1(C(c2ncc3ccccc3n2)C(=O)NC)CCCCCC1C1CCCO1 c1(CNC(CN(C(=O)C(F)n2ccnc2)CC#C)=O)cc(C)cc(Cl)c1 c1(CN2CCCC(O)C2)cc(Cl)c(Br)cc1Cl C1(C(=O)NC(C(=O)NCC=CCCC)CC2CCOCC2)CCOCC1(C)C Cc1ncc(Cl)c(C(N2CCC(N(C)C(c3ccc(C4CC4)s3)=O)C(C)C2)=O)n1 C(CNC(C1(C#N)CCCO1)=O)(C(C)(C)C)NC(c1nc(C(C)C)sc1)=O Cc1ccc(-c2nc(-c3ccnn3C)nn2-c2c(C)noc2C)c(F)c1F C1(F)(CNC(=O)C=Cc2cc[nH]n2)CCN(C(c2cc(Cl)no2)=O)C1 C1(NC(CC(CCC)C)=O)CC2CN(C(=O)CSc3ccccc3)CC2C1 c1(C(N2CCC(N(C)Cc3onc(C(C)OC)n3)C2)=O)cnc2[nH]cnc2c1 CC(C)(C)CC(=O)NC1CCOC1C(=O)Nc1ccccc1SCCO CCCC(C(=O)N(CCCCNC(=O)C(N)=O)C)OCc1ccccc1 C1(C(=O)NCC(C)NCc2cnc(O)c3ccsc23)CC(c2cnn(C)c2)=NO1 CC1CN(C(C2(C)CC(F)C2)=O)CCC1CNC(C1CCCC1)=O c1(C(N(CCn2cc(C(C)O)nn2)C)=O)cccc(N(C)C(C)C)c1 N1(C(C2N(CC)CC2)=O)CCC(c2cc(CNC(=O)C(O)CC(=O)OC)on2)CC1 c1(NC)cccc(C(=O)NCC(F)CNC(=O)CN(C)C(c2ccccc2)=O)n1 C1(NC(C(C2(O)CN(C(c3c[nH]c(=N)o3)=O)C2)F)=O)CC2CCCN2C1 N1(C(CCCC=C)=O)CCC2(CC2NC(C23CCC(C2)C3(C)C)=O)C1 C1(NC(C2N(C(=O)NC)CCC2)=O)CCCCC1NC(c1ccc(Cl)cn1)=O N1(C(C(C(C)(C)C)OC)=O)C2CCC1CC(NC(C1CCC1(C)C)=O)C2 Cc1cnc(CNC(=O)C(C)(C)NC(=O)CC2CCOC2)nc1 C(=O)(C(CCC(C)C)NC(C1CC(=C2CC2)C1)=O)N(C)CC1(CC)CCC1 C=C(C)CC(C)C(=O)NCC1CCN(C(c2cnc(C)n2C(F)F)=O)CC1 C1(CNC(C2CC(=C)C2)=O)CCCCN1C(C1CC(OC)(OC)C1)=O C(N=c1ccnc(NC2CCCC(F)(F)C2)[nH]1)c1cncc(C)c1 Cc1ccc(NC(=O)CC23N(C(CCCCNC(=O)C(C)C)=O)CC(C2)C3)cc1 C(=O)(CCC(O)C(C)(C)C)NCC1(CNC(c2c(OC)nn(C)c2)=O)CC1 N1(C(=O)NCCNS(N)(=O)=O)CCOC2(CC1)CCS(=O)(=O)C2 C1(CNC(c2scc(C)c2)=O)CCC(C)(C)CN1C(C1CCCN1C1CC1)=O c1(C(=O)NC(C2CN(C(CC(CC)SC)=O)C2)C)ccc(O)c(F)c1 CN1CCS(=O)(=O)CC1CC(=O)NC1CCCC1NC(c1cncc(N)n1)=O C1(CC=C)(NC(c2nc(Cl)cs2)=O)CC2CCC(C1)N2C(=O)C(CO)N(C)C Cn1cc(CNC(=O)OC(C)(C)C)c(CNC(C2CC2(C)C(F)F)=O)n1 C1(CC)CCN(C(=O)CNC(C2CC2C)=O)C1CNC(c1c(C)ncn1C)=O c1(OC)ccc(CCC(=O)NC(C)C(C)(C)NC(=O)CN2CCCCC2)cc1Cl N1(C(C=CCC)=O)CCN(C(c2ccc(C(C)C)c(F)c2)=O)CCC1C C(C(CO)N=c1nc(C(F)(F)F)[nH]s1)NC(C1(N(C)C)CCCC1)=O C(=O)(C(O)CC(N)=O)NCC1C(CC(=O)NCCCCC2C(C)C2)C1 N1(CC)CC(C(=O)NC2CCC2NC(=O)Cc2cccc(F)c2)CCC1=O C12CCCN(C1)C(=O)CC1(CC1)C(=O)N2.C(=O)(C(C)C1CC1)NCC1CC1.CCO c1(NC(Cn2c(C)cc(C3CC3)n2)=O)cccc(C=CC(=O)O)c1 c1(NC(c2ccccc2F)=O)ccc(Cl)cc1Cl CN1CCN(C2CCCN(C(C3CCC(C(N4CCCC4)=O)O3)=O)C2)CC1 c1(C(N2C3(CNC(CNC(C)=O)=O)CC(C2)C3)=O)cnc(C)c(C#N)c1 c1(C(C)(C)C)cc(N2CCC(OCCNC(c3ccoc3Br)=O)C2)ncn1 N1(C(C2N(C(CC)=O)C3CCC2C3)=O)CCCN(CC)C(=O)C1 C(CC(C(=O)N1CCCC(CN(C)CC)C1)NC(C1CN(C(N)=O)C1)=O)=CC C(C(COC)CC(=O)NC1CC(NC(=O)C(C(C)(C)C)OC)C1)OC N1(C(=O)CSc2n[nH]c(O)n2)CCC2(C(=O)NCC3(CCO)CC3)CC2C1 C#CCCCCCC(=O)N1CCC(C(=O)NCc2noc(COC)n2)C1(C)C N1(C(C(c2cnccn2)C)=O)CCCC(N(C(=O)Cc2n[nH]c(=N)s2)C)C1 C(=O)(CCC(C)(C)C)N(C)CC1CCCN(C(=O)CC2COCCO2)C1 CC1=NOC(C)(C(=O)N(CCC(=O)NCCN2CCCCC2C)C)C1 C(N=c1nc2ncccc2c[nH]1)c1cccc(CNC(C(C)(C)OCC)=O)c1 c1(OC)cnccc1C(=O)N(CC(C)NC(=O)C(C)(O)CF)C CCC(C)(CNC(=O)C(COC)N(C)C)C(=O)NC1(CCCCO)CC1 C1(C(=O)NCC2(CO)CC(C)(C)C2)CCOCCN1C(c1ccoc1)=O c1(OC(C)C)ccccc1NCC(O)CNC(=O)Cc1ccsn1 Cc1ncccc1CCC(N1CC(c2cnn(C)c2)C(N)C1)=O CC(Cn1ccnc1)C(=O)NCCCCNC(=O)C(=O)NCC(F)(F)F C(=O)(C(C)CC(C)C(C)=O)N1C(NC(CC(CCCC)OC)=O)C(OC)C(OC)C1 C(C(N=[N+]=[N-])C(=O)NC1C(C(N2CCC(CC)(CO)CC2)=O)C1(C)C)OCC C(=O)(C(CC(F)F)NC(=O)CP(C)(C)=O)N1CC(C(C)(C)C)OCC1 Cc1nc2c([nH]1)CC(C(N1CCSCC1CCO)=O)CC2 C1(NC(c2c(CNC(c3cc(CCC)[nH]n3)=O)cnn2C)=O)CN(C)CC1(C)C c1(C(CC(=O)N(C)CC2CN(C(COCC)=O)C2)C)cccc(OC)c1 C(C(C)C(F)C(=O)NCc1ccon1)NC(c1c(CC)nns1)=O c1(N(CC(CC)C)C)nc(N(C)CC2CCCO2)nc2ccccc12 N1(C(c2c(C)cc(C(F)F)o2)=O)C2CCCC1CN(C(=O)CC1CCOC1)C2 C12(NC(c3c(Cl)cnc(C)n3)=O)CCCN(C(=O)C(C)CC(N)=O)CC1C2 c1(NC(CC2CCN(C(c3ccc(C(N)=O)cc3)=O)CC2)=O)cnnc(Cl)c1Cl Cc1cnc2cccc(C(N3CC=CC(NC(=O)CC4(C)CC4(Cl)Cl)C3)=O)n12 C(C)(CC(=O)N(C1CN(C(c2c[nH]nc2Br)=O)C1)C)OC CCCCC(C)C(=O)NC(c1ccccc1F)CNC(=O)C(c1ccnn1C)O C(CCCC(CO)NC(c1cnn(C(F)(F)F)c1)=O)NC(=O)Cn1cnnc1O C1(C)(NC(=O)Nc2ccc(Oc3c(O)ccc(C)c3)cc2)CC(C)(C)OC1=O C=C(C)CCCC(=O)NCC(C1CCC1)NC(=O)C(C(C)(C)C)SC C12(NC(c3cnsc3)=O)CCCC(CN(C(c3ccc(C(F)(F)F)[nH]3)=O)C1)C2 c1(C(=O)Nc2ccc(Oc3cncc(F)c3Br)nc2)ccc2cnccc2n1 C(=O)(CCCC(C)(C)C)NC(C1CCCN1C(c1c[nH]nc1-c1ccoc1)=O)C CC(C)C(O)CC(=O)N1CCC(NC(=O)CCc2ccsc2Cl)C1 n1(CC)ccc(C(=O)NCC=CCNC(C2CCC2c2nc[nH]n2)=O)n1 c1(C(=O)NCC(C2CCN(C(C3CCCS3(=O)=O)=O)CC2)C)ccnn(C)c1=O C1(C(=O)OC)CC(N(CC(=O)NC(=O)CCC2CC2)C)CS1 N1(C(C2CCN(C(COCCOC)=O)C2)=O)CCCC(O)(CO)C1 c1(C(=O)OC(CCC)C)cc(Br)c(C)cc1Br C1(C)(C(C)C)CN(CC(=O)N(CC(O)C2CCC2)C(C)C)CCO1 C1(CNC(c2cc3n(n2)CCO3)=O)CC2(CCC2)CN1C(=O)CCOC1COC1 CC(F)(F)C(Cl)CN(CCO)Cc1ccc(C=CC(=O)OC(C)(C)C)o1 C(CCC(C(=O)NCCOCCSC)NC(=O)C(F)C1CCC1)OC C1(OC)CC(NC(c2cc(C)ncn2)=O)CN(C(C2CC2Br)=O)C1 CC(C)(O)C(F)C(=O)N(C1CCCC2(CC2)C1)C1CC2CCC1C2 C1(NC(CCN(C)CC)=O)CCCC(NC(c2c(C(F)(F)F)cnn2C)=O)C1 CC1(C)CCC(C(=O)NCC2(CNC(C3(N(C)C)CCC3)=O)CCC2)CC1 Cc1nc2ncccc2cc1C(=O)N(C)CCNC(=O)C(c1ccc(Cl)cc1)C c1(CN(C(CF)CF)C)cc(Br)c(O)cc1F CC1(C)CN(C(C2CCCC2CF)=O)CC(CNC(=O)COC2(C)CCCC2)O1 c1(CNC(C(N2CCCCC2=O)C)=O)cnc2[nH]c(O)nc2c1 N1(C(c2cc(C#C)cc(Br)c2)C(=O)NCCSC)CC2(CCC2)CCC1CO CC(C)CCC(C(=O)NC1CN(C)C(C)(C)C1)NC(C1CC(=O)C12CCC2)=O n1(CC(=O)NC2(CN(C(C(CC)SC)=O)C)CC2)nc(C(F)(F)F)c(Cl)c1C c1(OCC)ccc(CCC(=O)NCC2CCCCC2NCC23CC(C2)C3)cc1Cl C(=O)(CCC(F)(F)Cn1cc(C(O)C=C)nn1)N(CCC=C)CC(=O)N(C)CC C(=O)(C(F)(F)Sc1cnn(C)c1)NCCN(C(=O)CCc1ccc(C)s1)CC c1(C(=O)O)cccc(CN2CC3CCC2C3)c1.c12cccc(c1)OC2 C1(O)(NC(CCCOCCOC)=O)CCN(C(=O)CNC(c2cnoc2C)=O)C1 C(c1ccccc1C)=CC(=O)NC1(C(=O)NC2C=CC(C(=O)NC)C2)CCN(C)C1 C1(CNC(c2ccc(OC)c(C)c2)=O)CC2CCC(C1)N2C(c1csc(Cl)n1)=O c1(C(=O)NC2C3(CN(C(C(=O)NCC)=O)C3)CC2)cc(F)cc(N)c1C.C1CO1 n1(C(C)C)cc(Br)c(C(=O)NCC2CN(C(=O)CC3(C)CC3)CCO2)n1 Cc1nc(C)n(CCC(N2CCC(NC(=O)CCCc3sccc3C)C2)=O)n1 c1(NC(Cc2nccc(-c3cc(C)nnc3)c2)=O)ccc(F)nc1F C1(CNC(C(C)OCC)=O)CCC(NC(=O)CN(c2ccccc2)CC)C1 N1(C2CN(Cc3c(OC4CCCC4)cccc3)C2)CC23CCCC2(COC3)C1 Cc1ccc(Cl)c(C(N2CCCC(CN(C(=O)CNC(N)=O)C)C2)=O)c1N C#CCCCCCCNC(C1CCCCN1C(c1ccns1)=O)=O CN=c1cc(C(N2CCC(CNC(=O)CCNS(C)(=O)=O)(OC)CC2)=O)cc[nH]1 Cc1cn2c(n1)C(CNCc1nc(Cc3cccc(Cl)c3)no1)CCC2 Cc1ccc(CCC(=O)NCC(C)(F)CNC(=O)CSCCC#N)s1 N1(C(c2c(C)nn(C3CCC3)c2)=O)CCOCC(NC(C2CCN(C)C2)=O)C1 C(=O)(CC(CC)CCCC)OC(N1CC2CC1CN2C(CC1(CC=C)CCC1)=O)=O c1(CC(N2C(CNC(CCc3n(C)cnn3)=O)CCC2)=O)ccc(F)cc1F N1(C(C2N(C(C(COCC)(C)C)=O)C(C)C2)=O)CC2C(C1)C2(C)C Cc1cc(C)c(C(=O)NCC(C(=O)NCC(C2CC2)N(C)C)N(C)C)s1 CC(CC(=O)NCC1CN(C(C2CCC=CO2)=O)CC1C(F)(F)F)P(C)(C)=O c1(C(=O)OC)cccnc1C(N1CC2CC1C2NC(C12CC(CC(F)F)(C1)C2)=O)=O c1(OC(C(=O)NCC(C)(CO)NC(=O)CC=C(Cl)Cl)(F)F)ccc(Cl)c(F)c1 C1(NC(C(C(CC)C)OC)=O)CCCN(C(c2cncc(SC)c2)=O)CCC1 c1(-c2c(C)ccnc2F)cc2cc[nH]c2cc1C(=O)Nc1ccc(I)cc1F C#CC(CC(C)(C)C)NC(=O)NC(c1ccccc1F)c1ccccn1 C12(C(=O)NCC3CC(OC)CN3C(=O)CN(C)CCOC)CC1COC2(C)C c1(C(N(CC(C)N(C(Cc2ccc(OC)cc2)=O)C)C)=O)ccc2c[nH]nc2n1 N1(C(c2cc(CCC)on2)=O)CCC(NC(c2c(Br)cnn2C)=O)C(C)(C)C1 N1(C(CC(CC)CN(C)C)=O)CC=C(C(C)(C)C(=O)NCC(C)(C)N(C)C)C1 c1(C(N(C(CCNC(c2c(C(C)C)nco2)=O)C)C)=O)cc2sccc2s1 N#Cc1cccc2c(C(N3CCCCC3c3cnco3)=O)c[nH]c12 C(C(C)C(=O)NCC(C)CN(C(=O)C=Cc1ccco1)C)OCC Cc1cccc(CN2CCCC2C(N2CCCC2c2nn[nH]n2)=O)n1 C1(C(=O)OC)CC(C(=O)NC2CCOC2C)N(C)CC(=O)N1.C1CCC1.CO c1(C(=O)NCC2(O)CN(C(C3CCCN3C3CC3)=O)C2)cnc(C2OCCO2)s1 Cc1cc(C(=O)NCC2(CNC(=O)CC3CCCC(C)C3)CCCC2)sc1C C(=O)(CCCCCNC(=O)C1=C(Cl)CCC1)N(C1CCN(C(C)=O)C1)CC#C Cc1cccc(C)c1CC(N1CCC(O)C(NC(C2CC=CCO2)=O)C1)=O c1(C(N2C(CC)CN(C(=O)C=Cc3ccncn3)CC2)=O)cc2nc[nH]c2cn1 C1(CNC(C(C(C)O)C)=O)C2CCCC1N(C(C1CCn3ncnc3C1)=O)C2 N1(C(C(C)(C)OC)=O)CCC2(CCCC2NC(=O)C(CO)c2ccccc2)CC1 C1(C(=O)Nc2c(CN(CC)CC)cccc2)CC2CCCCC2O1 c1(C(N(CC)CC2CCCN2C(=O)CC(O)C(C)C)=O)noc2c(F)cccc12 C1(NC(c2c(C)nc(C3CC3)nc2)=O)CN(c2nnc(C)s2)CC2(CC2)C1 C=CC(C)C(C)C(=O)NCCC(=C)CNC(=O)CCSCCCC c1(CCNC(C2(CNc3cnc(C(=O)O)s3)CCCCC2)=O)ccc(Cl)cc1 CC1(C)CC(CNC(c2c[nH]nc2-c2ccccc2F)=O)CN1C(C1CC1F)=O C(=O)(C(F)C(F)(F)F)NC1C(NC(c2cc(CN(C)C)on2)=O)CCCC1 c1(C(=O)NCC(CCNC(C2CCC(C)O2)=O)O)c(C(F)F)cccc1F N1(c2cc(NCCCOCCCC)ncn2)CCN(C)C2(CCC2)C1 N1(C(c2ccc(C#N)c(Br)c2)=O)CCC2(CC1)CCN2C(c1ccnnc1O)=O Cc1cc(=NCc2ccncc2N)[nH]cc1S(=O)(=O)N(CCCF)C C=CCCCCCC(=O)N1CC(n2cc(CNC(c3n[nH]c(C)c3Cl)=O)nn2)C1 Cc1cc(Cl)nc(N)c1C(N1CC(NC(=O)C(C)(C)n2cnnn2)C(C)C1)=O C1(NC(c2c(COC)onc2)=O)CN(C(=O)CCNC(=O)OC)CC1C1CC1 Cc1cn(C)nc1C(=O)NCC1CCN1C(=O)C(C)(C)c1cnsc1 CCCC(CNC(=O)C(C)OCCC(C)C)C(=O)NC(c1nccs1)CC CC(C)CC(C(=O)NC1CCCSCC1)NC(c1ccns1)=O C(=O)(C1CCCCc2ccccc21)N1CCC(O)(CNC(C(C=C)(C)C)=O)C1 C#Cc1cccc(C(=O)NC(C)CNC(c2nc(CC)oc2C)=O)c1Cl C12(NC(=O)CC3CCCC3)CCC(NCC3CC4CC4C3)(CC1)C2 c1(CNC(C2CCCC3CNCC23)=O)cccc2c1OCCCO2 N1(C(C2(CCCC)CCC2)=O)CCCC2(CC(NC(c3cc(C)sn3)=O)C2)C1 C(=O)(C1Cc2ccccc21)NCCCCCN(C)C(C1C(F)(F)C12CC2)=O C1(NC(c2c(CC(C)C)n(C)nc2)=O)CC2CC1N(CC=Cc1ccccc1)C2 N1(C(c2cc(C)sc2NC)=O)CC2CC1CN2C(c1ccc(I)cc1Br)=O Cc1ccncc1NC(=O)C(C)NC(=O)C(C)(O)Cc1ccccc1 N1(Cc2cc(C(C)(C)C)[nH]n2)CCN(C(=O)Cc2ccco2)CC1C1CCC1 C=C(C)CN=C(NCC(C)(C)F)NCc1ccc(C(C)(C)C)nc1 C1(CNC(C(c2cnn(C)c2)C)=O)CN(C(c2nc(Cl)c(Cl)s2)=O)CC1O c1(Cc2cn(CC(C(N3C(C(=O)O)C(O)CC3)=O)O)nn2)ccc(F)c(F)c1F.C C(=O)(CCCC(=O)NC(c1ccc(N(C(C)=O)C2CC2)s1)=O)NC(CCC)C c1(C(=O)NCCCC(C)NC(=O)C(N2CCNC2=O)C)ccc(NC=O)cc1 C(=O)(C1=COCCO1)N(CC(C)N(C(CCc1cc(C)on1)=O)C)C c1(NC(C)=O)ccc(S(=O)(=O)N2CCOC(Nc3cccnc3C#N)C2)cc1 C1(C)(n2c(N(C)Cc3c(C)cccc3)nnn2)CCCN(C(C)(C)C)C1 c1(CNC(CC(CNC(CC2CC(OCC)C2)=O)O)=O)ccc(F)c(C)c1 C12(NC(c3ccc(CC)o3)=O)CCC(C1)N(C(c1c(C)nsc1C(=O)OC)=O)C2 Cc1ccc(C)c(-n2cc(NCCN(C)CC3CCOCC3)nn2)c1 C(=O)(N=c1cc2n([nH]1)CCCNC2=O)N1C(C)C2CC1C2 C1(CNC(C2C(C)=C2)=O)CN(C(c2ocnc2C)=O)CCC12CCOCC2 CC1(C)CCC(F)(F)CC1C(N1CC2CCCC(C1)N2C(C1CC(F)(F)C1)=O)=O c1(SC(=O)OC(c2cn(CC)nc2)C)cc(OC)ccc1[N+](=O)[O-] N1(C(c2ccc(CC(=O)OC)[nH]2)=O)CCN(C(C2OCC2(C)C)=O)C2(CCC2)C1 N1(C(C(c2n(C)ncc2)O)=O)C2CCC(C2)C1CC(=O)NCC(=O)NCCO Cc1ccccc1CC(N1CC(F)CC1CNC(c1cn(CCF)nn1)=O)=O C=Cc1cc(-c2ccc(C(CC(=O)OC)NC(=O)C3CC3)s2)cc(F)c1 C1(CNC(C2(C)COC2)=O)CC2(CCN(C(=O)C=Cc3cccs3)CC2)CO1 C1(C(N(C2CCN(C(CC=C=C)=O)C2)C)=O)CN(CC(F)(F)F)CC1C C1(CNC(C2CN(S(C)(=O)=O)C2)=O)C=CC(CNC(=O)CCc2cccn2C)C1 c1(NCc2cnn(CCC)c2C)ncc(C2=COCC2)cn1 c1(C(=O)OCC)nc2[nH]ccc2c(=NCC(CCOC)Oc2ccccc2)[nH]1 Brc1ccc(C(c2nnnn2C2COC2)NC2C3COCC23)c(C(F)(F)F)c1 C1(NC(c2c(C)ncs2)=O)CCC2CN(C(=O)CCCOC3CC3)CCC2C1 CCCC(CC(C)C)C(=O)N1CCC(C(=O)N(C(C)CC(C)C)C)C(C)C1 Cc1cccnc1C(=O)NC1CN(C(=O)CC2(C)CC2(Cl)Cl)CC1C(F)F C(=O)(C1=NOC2(CCC2)C1)NC1CCN(CCCNC(CC=C(C)C)=O)C1 Cc1nc(NC2CCN(C(C3CCCCS3)=O)C(C)C2)cc(C#N)n1 c1(NCC(C)N(C(C(CCC)c2ccccc2)=O)C)cccc(F)c1C#N c1(C2(CNC(=O)N(C3CCCC3)CCO)CCCC2)cccc(F)c1F CC(C)(CC(=O)NCC1CC(O)C(O)C1)NC(=O)Cc1cccnc1F N1(C(c2cc(CCC)[nH]n2)=O)CC(C)C(NC(=O)COCC2(F)CC2)C(C)C1 c1(C(=O)NCCC(C)CCNC(C2CNC(=O)N2)=O)ccc2[nH]ccc2c1F Cc1cnn(C)c1C(=O)N(C)CCNC(c1n[nH]cc1C1CC1)=O c1(CC(=O)NC(CCCC)CNC(=O)C(C)O)ccc2[nH]ccc2c1 N1(C(C2C(c3c(C)occ3)C2)=O)CCC(C2CC2)(CNC(=O)CCS(N)(=O)=O)C1 C1(CNC(CCCC(=C)C)=O)N(C(c2cc(C3CCC3)[nH]n2)=O)CCCC1(C)C c1(C(N2C(CC(=O)NCc3ncc[nH]3)COCC2)=O)ccc([N+](=O)[O-])cc1F C1(C(=O)NC(CNC(CCCC2C(C)C2)=O)(C)CO)CC2(CCC2=O)C1 Cc1ccn(CCC(=O)NCCCC(C)NC(C2COC(=O)C2)=O)n1 N1(C(c2c(CC)cco2)=O)CC2CC1CN(C(=O)CC1OCCC1(C)C)C2 C12(CNC3(C)CCN(C(=O)OC)C3)CCCC(CO1)C2.C12CN(C1)CC(=O)N2 C(CSC)(C(=O)NC1C=CC(CNC(C2(C)CC2C)=O)C1)OC C1(CNC(C(CCCC)C)=O)CC2(CO1)CN(C(=O)C=C(C)c1cccs1)C2 C1(C#N)(C(=O)NCCCCN(C)C(C2CC(=O)CC(=O)N2)=O)CC2CC2C1 C1(C(=O)NCc2csc(C)c2C)CCC(C)(C)N(C(=O)Cc2ncccc2F)C1 N(C(=NCc1cccs1)N1CCC2(CCOCC2)CC1)C1CC2C(=O)C(C1)CC2 C1(O)(CN(C(CC2ON=C(C)C2)=O)C)CCN(C(C2(C)CC2)=O)C1 N1(C(C=Cc2c(C)ncs2)=O)CCCC(F)(CNC(C2(C)CC2(F)F)=O)C1 c1(CC(=O)NC2CC3CCC(C2)N3C(C23COCC2C3)=O)coc2ccccc12 C(=O)(C1=CCCCCC1)NCC(C1CCC1)NC(C(SC)SC)=O Cc1cc(F)cc(C)c1C(N1CC2C(CNC(C3(C)CC3C)=O)C2C1)=O C=CC1OCCCC1C(=O)NCCOC1CN(C(=O)CCc2csc(=N)[nH]2)C1 N1(C(CS(=O)(=O)NC)=O)CCN(C(=O)CCC(C)(C)[N+](=O)[O-])C2CCCCC12 C(=O)(C(CNC(=O)CNC(=O)C(C)CC)C(C)C)N(C1CCOC1)CC#C C=C(C)C(CC(=O)N(C(C)CNC(c1coc(CCC)n1)=O)C)OCC N1(C(CCC(C)N(C)C)=O)CCC(NC(=O)C=Cc2ccc(F)cc2)C1(C)C C1(C(=O)NCC2(CNC(C3(F)CCCCCC3)=O)CC2)CCC2C(C1)C2(F)F CC(C)CC(F)(F)C(=O)N1CCN(C(=O)CC2(O)CCCCCC2)CC1C(C)C CC(C)(C)CCC(F)C(=O)NCC1CN(C(=O)C(C)(C)C)CC1C1CC1 Cc1cnn2cc(C(N3CC4CC(NC(=O)Cn5nnc(=O)[nH]5)C3C4)=O)cnc12 C1(C(=O)NC2CC(NC(C3CC(CN(C)C)C3)=O)C2)(C(F)F)CCCO1 S(=O)(=O)(c1cccc2c1COC2=O)N(C)CC1CCN(C)C1 c1(NC)ncccc1C(=O)NC1CC(C(F)C(=O)N(CC(C)C#N)C2CC2)C1 C(=O)(C1=CCCC1(C)C)NCCN(C(=O)CC(C)(F)F)CCc1nc(C)sc1 CCCC(CC(C)C)C(=O)N1CCCC(O)(Cn2cc(C(O)C(C)C)nn2)CC1 n1(CCC(=O)NCC2(C(N3CCC=CC3)=O)CC2)ccccc1=O.C1CS1 c1(CC(=O)N(C2CN(C(=O)COCCn3nccn3)C2)C)ccnn1C C1(C(N2CCC(NC(COc3ccn(C)n3)=O)C2)=O)CCc2nnnn2C1 Cc1ccccc1CC(=O)NCC1(NC(c2cc(O)ncn2)=O)CCC1 C(CN=C(NCc1ncnn1C)N(C)Cc1cc(CC2CC2)nn1C)OC C12(OC)CCC(C(=O)NC34CC(NC(c5ccc[nH]5)=O)(C3)C4)(CC1)C2 C12(NC(C(CSC)OC)=O)CN(C(=O)CC(F)F)CC1CS(=O)(=O)C2 C1(C(=O)NCc2c(C)scn2)CCN(C(=O)CC(C)(C)O)C12CCC2 C=CC1(NC(=O)C(CNC(c2cccnc2S)=O)OC)CCOCC1 Cc1[nH]c2ccc(Cl)cc2c1C(=O)NOCC(N1CC(n2ccnn2)C1)=O c1(C(=O)NCC(CCCC)NC(C2CC2(C)Br)=O)ccc(C)c(C)n1 c1(C(=O)Nc2scc(COC)n2)cc(I)ccc1[N+](=O)[O-] C1(CC)C(NC(C2CCCN2C)=O)CCCN1C(c1cccc(=O)o1)=O c1(C(N2C(CNC(=O)C=CC3CCCC3)CCC(C)C2)=O)cccn2nccc12 c1(C(N(CCCCNC(C2C(C)(C(C)C)C2)=O)C)=O)ccc2cnccc2c1 Clc1ccccc1C=CC(=O)N(C1CC1)Cc1cncc(Cl)c1.C1(O)CCSCC1 C(N=c1[nH]c2ccc(F)cc2s1)C1CCC(NC(CC2(O)CCCN(C)C2)=O)C1 N#Cc1ccnc(NC2CN(C(C3CCC(CO)CC3)=O)C2)n1 C(=O)(CC(C)CC(=O)OC)NC1CC=C(C(=O)NCCC(CCC)C2CC2)C1 Fc1cc(CNC(c2nnnn2C2CCOC2)c2cnn[nH]2)cc(Cl)c1 C(=O)(C1=C(Cl)CCOC1)NCC1(C)C(C)CN(C(CC2CC(=C)C2)=O)C1 C1(CNC(C2C3C(=O)OCC23Br)=O)CC2(CC2)CN1C(c1cc(O)nc(Cl)c1)=O C1(CNC(C(C)OC)=O)CCC(C(=O)NCc2cc(C)[nH]n2)O1 c1(CC)ccc(N)c(C(=O)N(CCCNC(C2CC(=O)N(CC)C2)=O)C2CC2)c1 Cc1cc(=O)c(C(N2CCCC(CNC(C3(C)CCCCC3)=O)CC2)=O)cn1C c1(C(=O)NCC(CC=C)NC(c2cccc(CC)c2)=O)cc2n(n1)CCC2 N1(C(c2[nH]cc(C)c2)=O)CCOCC1CCNC(c1cccnc1C(F)(F)F)=O C1(NC(CC)=O)CCC(NC(=O)C(F)CC2CCCCC2)C1 C(=O)(C(C)CC(C)(C)C)NCC(CCC)C(=O)N1CCCN(C(N)=O)CC1 C(C(C)(C)C#CC(=O)NCc1ncccc1O)NC(C(C)c1ccco1)=O c1(C(=O)NCCN(C(CC(CC)C)=O)CCOCCO)nc(C)n(C)c1C Cc1cc(=N)[nH]cc1C(=O)NC(C)(C)C(C)NC(c1cc(Cl)sc1Cl)=O Cc1ccc(C(=O)NC2CC(C)N(C(=O)CCOC3CCCC3)C2)cc1[N+](=O)[O-] c1(NCc2ccc(C(=O)OC)s2)cc(Cl)ccc1[N+](=O)[O-].N12CCC3(CC3C1=O)C2 C1(NC(CCCC(=C)C)=O)CN(C(C2CC3CCCCCC23)=O)CC2(CCC2)C1 CON1CCC(C(=O)NC2(CO)CN(C(c3cnccc3N(C)C)=O)C2)CC1 Cc1cc(C(=O)NCC2C(CNC(=O)C(C(C)C)n3cccc3)C2(F)F)c(C)s1 N1(C(C2(C)CC(C)(C)C2)=O)CCCC(C2CCCN(C(=O)CSC(=N)N)C2)C1 c1(CC)c(OC)cccc1C(=O)N(CC(CC)NC(c1ccnc(S)c1)=O)C C(CCC(O)C(=O)NC1CC(=O)NC1(C)C)NC(CC(C)N(C)C)=O C(=O)(CCC#Cc1ccccc1)NC1(CNC(C2C(C=C)OCCC2)=O)CC1 n1(CC)nc(C)cc1NC(C12CC1CN(Cc1ncccc1C)C2)=O C(=O)(CCC(C)SC)NCCC(c1cccs1)N(C(C1C(C)=C1)=O)C c1(C(=O)NC(C(=O)NCC(C)(O)C2(C)CC2)c2ccco2)cc(CO)oc1C C1(NC(CSCC)=O)C2CC3CN(C(c4ccc(=O)n(CCF)n4)=O)C1C3C2 c1(-n2c(C(=O)NCC3(CCNC(C(CSC)O)=O)CC3)cnn2)ccccc1F CC1(C)C(=O)CC1C(N1CCCC1C=CC(=O)NCC1(C2CC2)CCCO1)=O C(CCCCC(=O)N1CCOC(C(N2CCCC(C)(N(C)C)C2)=O)C1)=CC c1(OC)c(Cl)cc(C(=O)NC(C)CCNC(c2cnc(=N)[nH]c2)=O)nc1Cl c1(CNC(C2CC(C)CN2Cc2ccccc2)=O)ccc2c(c1)C(C)C(C)O2 S(=O)(=O)(c1ccccc1)N1CCC(C(=O)NCC2OCC(=O)NC2)(CO)CC1 C1(NC(c2c[nH]c(=N)s2)=O)C2CC3CN(C(c4ccnc5[nH]cnc45)=O)C1C3C2 C(=O)(CCC(F)(F)C(F)F)N(CC(CC)NC(c1cncc(N(C)C)c1)=O)C c1(CNC(CCN(C(=O)C(O)C2CCCC2)CC=C)=O)c[nH]c(=O)cn1 Cc1c(C(=O)NC2CC(NC(c3ccon3)=O)C(O)C2)sc2ccsc12 Cc1c(C(N2CCCC(N(C(=O)CC(C)F)CCF)C2)=O)sc2cccc(F)c12 C1(C(=O)Nc2c(C)ccc(C)c2)CC(N=c2cc(C(F)(F)F)nc(Cl)[nH]2)C1 Brc1ccc(CC2N(CSCCC3CC3)CC2Cl)cc1 c1(C(=O)NCCN(C(=O)CC2CS(=O)(=O)C2)C)csc(-c2cnn(C)c2)n1 N1(C(C(C)=CCC)=O)CCCC1C(=O)NCC(C)(C)COC C1(OC)CC2(C1)CC(NC(=O)C=C(C)CNC(C1(C)CC1C)=O)C2 C1(NC(C(C)=C2CCCC2)=O)CCCC(CNC(c2ncn(C(C)C)n2)=O)C1 N1(C(C(CC)N(C(C)=O)CC)=O)CCC(C)(C(N2C3CNCC2C3)=O)C1 c1(NC(C(C2CCOC2)NC(c2cc(CC)[nH]n2)=O)=O)ccc(CCO)cc1 C1(CCNC(C(CCSC)O)=O)CCCN(C(c2cc(Cl)c(C)cn2)=O)CC1 CCCC(C(=O)NCC(c1ccco1)O)NC(=O)C(C)(C)CC1CC1 N1(C(C(C)(C)CC(F)(F)F)=O)CCC2(CO)CN(C(=O)C3=CCCCC3)CC2C1 c1(C(=O)NCC(C)NC(C2(F)CC=CC2)=O)cc(N)cc(O)n1 S(=O)(=O)(c1cc(C(F)(F)F)cc(Cl)c1)N1CCC(C(N(C(C)C)C)=O)CC1 N1(C(Cc2scc(C)c2)=O)CCCC(C2CN(C(=O)CSC3CCOC3=O)C2)C1 C1(C2(NC(=O)COC3CCCC3)CC2)CCCCN1C(C1CC=CCO1)=O Cc1cc(N2CCC(c3nc(C)no3)C2)nc(=NCC=C2CCC2)[nH]1 c1(C(=O)NCC2(CNC(c3nccs3)=O)CC2)cc(C(F)F)ccc1Cl c1(CC(C(=O)N(C)Cc2nncs2)NC(=O)CNC(N)=O)cnn(C)c1O c1(NCC2CCN(C(=O)NC(=O)OC)CC2)c(C)cc(CC2CC2)nc1O c1(CC)cc(C(=O)NC(CNC(=O)Cc2csc(C(C)(C)C)n2)C(C)C)nn1C c1(C(N2CCC(CC=C)(C(=O)NC(C)C(C)C)C2)=O)cc(C)cc(C)c1 S(=O)(=O)(c1cccc2nonc12)N(C1CNC1)C(c1nnc(-c2ccco2)o1)=O c1(CC(=O)NCC(CC=C)NC(=O)CCC(F)(F)F)coc2c(C)c(Cl)ccc12 n1(CC=C)cc(C(=O)NC2CCN(C(c3cc(-c4ccccn4)c[nH]3)=O)C2)nn1 C(=O)(NNc1cccc(C(F)C(F)(F)F)n1)c1c(F)ccc(C(N)=O)n1 C1(C(N2CCC(C(=O)OC)C2C)=O)CCN(C(=O)CCc2nccs2)C(C)(C)C1 c1(OC)ccnc(OC)c1C(=O)NC(C)C(C(C)C)NC(c1ccccc1O)=O CCCCCCC(F)C(=O)N1CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1 c1(C(N(C2CN(C(c3cccc(OC)c3)=O)C2)C)=O)cc2c(O)cccc2[nH]1 C12(CNC(c3ccc(C(C)(F)F)cn3)=O)CC(NC(=O)C(C)(C)CO)(CCO1)C2 c1(CN2C(C(=O)NCC3CCOCC3)COCC2)cn2cccnc2n1 c1(OC)ccnc(F)c1C(N1CCC(O)C(NC(c2cc(F)ccc2F)=O)C1)=O C(=O)(C1=CC2C=CC(C1)C2)NC(C1(O)CCN(C(=O)CCc2ccncn2)C1)C C1(C(N(C)CC2(O)CN(C(=O)CC(C)(F)F)C2)=O)CC2(CCC2)CO1 C(C)(C(=O)NC1CCCC1NC(C1(CCOC)CCCC1)=O)(C(C)C)OC CN1CCCCCC1C(=O)NC1(CO)CCN(C(=O)CCCC2CC2)C1 Cc1cnccc1C(C)C(=O)NC1CCCC(NC(c2ccc(=N)[nH]c2)=O)C1 CCC(CO)(C(=O)NCc1cccc(CNC(c2cccc(NC)n2)=O)c1)OC CCC(CC(=O)N1C(C(=O)N(C)CC)CC1C)NC(=O)COC(C)=O N1(C(C2CC(CC)C2)C(=O)NC(C)(C)C)CCS(=O)(=O)C2CCCCC12 C(=O)(C1SCCc2sccc21)NCC1(OC)CCN(C(=O)CCSC)CC1 c1(C(=O)NCCC(C)N(C)Cc2cccc(F)c2F)cccn2ccnc12 c1(C(N2CC(NC(c3c(OC)nn(C)c3)=O)(CF)C2)=O)cccc(C)c1F C1(CNC(=O)NCc2csc(C3CC3)n2)OCC2CCC1C2 c1(C(=O)NCC2CC(NC(C3C(C)(C(C)C)C3)=O)C2)ccc([N+](=O)[O-])c(O)c1 N1(C(C2C3CC4C(C3)C24)=O)CCC2(CCN(C(C3(C4CCCCO4)CC3)=O)CC2)C1 N1(C(Cc2c(C)cccn2)=O)CCCN(C(=O)CC23CCC(CC2)C3)CC1 C1(C(N2CC3C(CNC(=O)COC4CCOC4)(C3)C2)=O)CCC2(CCCCC2)C1 C1(CNC(c2cc(C)no2)=O)(NC(c2cc(=O)n(C)o2)=O)CCCCC1C CCC(C(C)CN(C)C)NC(=O)C(CC1CC1)NC(=O)CN=[N+]=[N-] C(CCCN=c1nc(N2CCC3(CC2)CC3OC)c2c([nH]1)CCOC2)OCC c1(OC)cc(N2CC3C(C(=O)Nc4ccccc4NC)C3C2)nc(OC)n1 CCC(CC(=O)NC(C1CCN(C(c2nc(C)nn2C)=O)CC1)(C)C)OC C(CCC)(C(=O)NC12CC(NC(=O)C(C3CC3)OC)(C1)C2)=CC c1(C(=O)NC2CCCC(N(C(c3c(C)nc(C)s3)=O)C)C2)c(C)oc(C)c1C c1(C(C(=O)NC2CN(C(C3CCCS3)=O)C2)OC)ccc(F)cc1 c1(NC(C2(C)CCN(C(COC(CC)C)=O)C2)=O)cccc(C#N)c1 C1(CNC(COCC(C)C)=O)CN2CCCCC2CN1C(c1ccc(O)cc1)=O c1(N2CCc3n(CC)cnc3C2)sc(=NCC(C)(C)NC(=O)OC(C)(C)C)[nH]c1Cl C1(COC)CCOCC1NS(=O)(=O)CCC1(c2nnc(C(=O)OC)o2)CCOC1 N1(C(CCOC(C)=O)=O)CCC2(CCC2NC(=O)CC2CCC(=O)O2)CC1 N1(C(CN(CC)CC)=O)CCC(CNC(c2occ3c2CCC3)=O)C(F)(F)CC1 Cc1cc(=N)[nH]cc1C(N1CC(O)(CNC(c2cnc(-c3cccs3)o2)=O)C1)=O C=C(C)CCCNC(=O)C(C)=CCNC(c1cc(C)sn1)=O C1(CCC)CN(C(c2cnn(C)c2Cl)=O)CCN1C(c1nc(CC)oc1C)=O C(C)(N=c1[nH]ncs1)C1OCCN(C(c2ccc(OCC)nc2)=O)C1 c1(C(=O)NC2C(NC(c3cn(CCC)nn3)=O)CC2)cn(C)c2c(Cl)cccc12 C1(C(=O)N(C2CC3CNC2C3)Cc2ccccn2)CCC2CNCCC2C1 c1(C(N2CC3CCN(C(c4cnn(C)c4F)=O)CC32)=O)cc2nn[nH]c2cc1F c1(C(COC)NC(C2CC2C#N)=O)ccccc1CNC(c1cc[nH]n1)=O C1(CCc2scc(C)n2)CN(CC2CNC(=O)O2)CCO1.c12cn(nn1)C2 c1(SCC)ccccc1CC(=O)NC(C)CNC(=O)C(n1cc(Cl)cn1)C c1(C(F)(F)F)cccc(CNC2CC23CCCC3)c1 C1(NC(c2cc(C)cc(O)n2)=O)CC2CCC1CC2NC(C1CCCOC1C)=O C1(NC(c2cc(C)no2)=O)CCC(NC(C2CC2(c2ccccc2F)C)=O)CC1 c1(NC(C2N(C(c3cc(OC)c(OC)nc3)=O)CC2)=O)cc(Br)ncc1[N+](=O)[O-] Cc1ncc2ccccc2c1C(=O)NC1(CCNC(=O)Cc2scnc2C)CC1 C(=O)(C(C)(C)CC(=O)N1CCSCC1CCNC(=O)C(C)c1cc[nH]n1)OCC C(=O)(C(C)CC(C)(C)C)NC1CN(C(C(CC)CC)=O)CC(C)C1 c1(-n2cc(C3CCN(C(C4CNC(=O)O4)=O)C3)nn2)cccnc1Cl c1(OC)cccc(C(N2CCC(F)C(NC(=O)CN(C)C(N)=O)C2)=O)c1F C1(C(N(CC#C)CCOC)=O)(CC)CCCN1C(c1cc(C)ncn1)=O c1(C(=O)NC(C)CNC(C2CCS(=O)CC2)=O)c(O)c2ccccc2n(C)c1=O Cc1c(OCC(=O)NC2CC(NC(C3COCC3(C)C)=O)C2)cccc1CO C(=O)(CCCCCNC(N)=O)NCC(CNC(C(c1cccc(Cl)c1)C)=O)O c1(N2C(CCCNC(C3CC(O)(CC#C)C3)=O)CCC2)cncc(C#N)n1 S(=O)(=O)(c1ccc(NC(c2ccc(-c3ccccc3)o2)=O)cc1)NC(C)C C1(N(C)C(=O)NCC2(c3cccs3)CC2)CCC(F)(F)CC1 N1(C(CCOCCN(C)C(C2(CCO)CC2)=O)=O)CC(F)(F)C1C1CC1 C1(O)(C(C)NC(c2cnsc2)=O)CCN(C(c2cncc(C(F)F)c2)=O)C1 C1(C(=O)NC)(CF)CCN(CC2CC2Br)C1 S1(=O)(=O)c2ccc(C#N)c(c2)N(C)CCCCN1C.C(C(C)OC)OC N1(C(C(=O)NC(c2cc(-c3ccc(F)cc3)nn2C)C)=O)CCCNC(=O)CC1 c1(C(=O)NCCC(C)NC(c2cncc(C(F)(F)F)c2)=O)cc2c(ccn2C)s1 CC(CN(C(=O)CCN(CCO)C(=O)OC)C)S(C)=O.C(C)(C)(C)O c1(CC)ccc(OCC(N2CCC(C(C)NC(C3CCCC3)=O)C2)=O)cc1 C(CCC)(CCCNC(=O)CN1CC(=O)NC1=O)NC(COCC#C)=O c1(SCCNC(=O)NCCNC(C)=O)ncccc1Cl c1(NC(C(=O)NCC(C(CC)C)=O)=O)cc([N+](=O)[O-])ccc1Br N1(C(c2conc2C)C(=O)NCCSC)CC(C)OC2(CCC2)C1 N1(C(c2occ(C)c2)=O)CCN(C(c2cnc(C(C)C)s2)=O)C(CC(C)(C)C)C1 Cc1nc2ccc(NC(=O)COC(c3cc(Cl)cc(Cl)c3F)=O)cc2[nH]1 N1(C(c2ccc(C#N)cc2)=O)CCN(C(=O)CC2CCC(C#N)C2)CC12CCC2 C1(C(=O)NCC(CN(C(Cc2cnc(C)[nH]2)=O)C)(C)C)CCn2c(cnc2C)C1 Cc1cnc(C)c(N2CCOC(C(=O)NC3CC(=O)N(c4ccccc4)C3)C2)n1 C1(C(=O)NC2(CC=C)CCN(C(C3CC(CCC)C3)=O)C2)CC2(CCCC2)C1 CN1CCCC(NC(C2CN(C(=O)C=Cc3ccsc3)CC2C2CC2)=O)CC1 C12(C(=O)NCC=CC(=O)NCC(C)SC)CC(F)(C1)C2 N1(C(Cn2nc(C)oc2=O)=O)CCC(CO)(CNC(C2CC=CCC2)=O)CC1 C1(C(CNC(=O)CCc2ccncc2)F)CCN(C(=O)CC2(COC)CC2)CC1 c1(SCC(C(=O)OCC)(F)F)nc(C2CC2)nc2cccc(F)c12 Cc1cc(CNC(=O)CN2CCCC2)oc1NC(=O)OC(C)(C)C C1(=O)C(CCC2CC2)N2CCN(CC2)N1.c1(SCO)cnc(C2CC2)o1.C(CC)SC c12cc(cc(F)c1)C(=O)N2.C1(C(=O)OC)(CO)CCCC1.C12CCC1C(=O)N2 N1(C(c2cc(C)nc(O)c2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC(C#N)C1 n1(CC(=O)NCCC(CNC(CCC(=C)C)=O)O)nc(C(F)F)c2c1CCC2 N1(C(C2C(C)CC(=O)N2)=O)CCCC(C2CN(C(=O)CC3C=CCC3)C2)C1 N1(C(CCC(CC)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(F)(F)COC c1(C(N2CCCN(C(CC3(C)CC3F)=O)CC2)=O)cc(F)c(Br)c(Cl)c1 C1(C2CC2)(C(=O)NC2CCCC2NC(=O)C(O)Cc2ccccc2)CCC1 C1(CNC(c2nn(C)c(Cl)c2)=O)CN(C(C2SC3C=CC2CC3)=O)CCCO1 N1(C(=O)C(F)(F)Cl)C(C(N2CCC3(CCOC3)C2)=O)CC2CCCCC12 C1(C(N2CC(O)(CN(C(C3N(CC)CC3)=O)C)C2)=O)COCC(C)O1 C1(C(=O)NCc2cc(C(N3C(C)(C(=O)NC)CC3)=O)on2)CC(=O)C1(C)C C(=O)(C(CC(C)C)NC(=O)C(C)NC12CCC(CC1)C2)OC CC(C)C(C(=O)NC(C)CNC(c1c[nH]nc1C(C)(F)F)=O)n1cncn1 C(c1ccc(C#N)cc1)=CC(=O)NC1CCC(C)N(C(c2cncnc2)=O)C1 CCC(CCC(=O)NCC1(O)CCC(O)CC1)OCC C1(OC)CN(C(C2(OC)CC2)=O)CC1C(N1CC(C)(O)C1)=O C1(C)(C(=O)NC2C(CCC)CN(C(=O)C(n3cc(C)cn3)C)C2)CC(=O)N(C)C1 C1(C(=O)NC2CC(F)(CNC(c3cnc(C(F)F)nc3)=O)C2)CCS(=O)(=O)C1 CC(C)CC(O)CC(=O)N1CCC(C(=O)NC2(C)CC(O)C2)C12CCC2 C1(C)(C(=O)NCC(C)CN(C)C(c2ncccc2C(C)(C)C)=O)CCCOC1 C12(C(=O)NC(CC(=O)NC(C)C)C)COC(C1)C(NC(c1nccn1C)=O)C2 N1(C(=O)NC2CCC2)CCCC(c2nnc(S)n2C2CCCC2)C1.C1S(=O)(=O)N1 C=CCC(C(=O)N1CC(OCC(=O)NCCC23CCCC2C3)C1)OC C1(CCCC)CCC(NC(C2(NC(=O)OC(C)(C)C)CC(CO)C2)=O)C1 Cc1ncc(C=CC(=O)NC23CC(CNC(c4cccc(F)c4)=O)(C2)C3)s1 N1(C(C(CC)C2CCOCC2)=O)CCN(C(=O)COC(F)(F)F)CCC1C C(=O)(C(F)(F)C(O)C(C)C)N(CCCN(C(C(c1c(C)nn(C)c1)C)=O)C)C C=CC1(C(=O)NCC(C)(C)CC(C)C)CCN(C(=O)CCN2CCCCC2)C1 C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1C2N(C(Cn3nnc(C)n3)=O)CC(CC2)C1 C1(NC(C=CC)=O)CN(C(C2CC3(C2)CC3F)=O)CC1N=[N+]=[N-] N1(C(c2c[nH]c(=N)s2)=O)CC2CC1CCC2NC(c1ccn2nccc2c1)=O N1(C(c2ccccc2CN2CCOCC2)=O)CCC(COCCOC)C(O)CC1 c1(C(N(CCCN(C(C(C)(C)OCC)=O)C)C)=O)nc(C)ncc1Cl C=CC1(C(N2CC(C)(F)C2)=O)CCN(C(=O)COc2ccsn2)CC1 C1(O)(C(C(=O)NC(C(C)CO)C)NC(=O)CCc2ccc[nH]2)CCCCC1 c1(C(=O)NCC2CN(C(CNC(C(C)C)=O)=O)C2)c(C2CC2)cccc1F C1(N(C(c2scc(COC)c2)=O)C)CCCN(C(=O)C(COC(C)C)OC)CC1 c1(C(N2CCC(O)C(C(N3CCOCC3CO)=O)C2)=O)c(Br)cccc1Br c1(C(=O)NC2(CF)CCN(C(C3CCC3(F)F)=O)C2)cnc(C2CC2)nc1O C1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)CCCC2)CCCCC(C)(C)C1 c1(C(=O)NCC(N(C)C(c2ncc(Cl)nc2Cl)=O)C2CC2)cccc2c1OCC2 C=CCC(CC(=O)NC1CC2OCCCC12)NC(=O)CCn1ccnc1C N1(CC(=O)NCC(CN(C(=O)CC2C=CCC2)C)O)C(=O)NC(C)(C)C1=O C1(CNC(C(CCSC)O)=O)CN(C(=O)C(C)(C)n2cnnn2)CCC12CCC2 C1(CNC(c2c(SCC=C)cccc2)=O)CCN(C(=O)CC(C)(C)O)CC1C N1(C(c2cncc(C=C)c2)=O)CCN(C(C2CCN(CC)C2)=O)C2CCC12 c1(OC)ncc(S(=O)(=O)NCCC(c2cccc(Br)c2)C2CCC2)s1 N(C(=NCCC(=O)OC(C)C)NC1CN(CC)C1)CC1OCCN(C(CC)C)C1 N1(C(C(Cc2cn(C)nc2)O)=O)CCC(CNC(=O)CCNC(N)=O)C12CCC2 Cc1cccc(C)c1OCC(=O)OC(C)(C)C.c12cccc(n1)NC(=O)NC2 c1(OC)ccc(C(N2CC(NC(=O)C(C3(O)CCCCC3)(F)F)C(F)C2)=O)cn1 Cc1cc(C#N)cnc1C(=O)NCCCNC(=O)CC1CS(=O)(=O)CCN1C CCCCCCCC(F)C(=O)NCC1CN(C(c2ccc(C)c(C)c2)=O)C2CC12 N1(C(c2cnc(COC)nc2O)=O)CCN(C(c2csnn2)=O)CC(C)(C)C1 C(=O)(CCC(=O)NCC1CCCN(C(=O)Cc2csnn2)C1)N(C(C)C)C c1(C(=O)NC2CC(F)(CNC(C3(CC=C)CC3)=O)C2)cc(Cl)cc2ccncc12 c1(C(=O)NCCC2(O)CN(C(C3CCC(CC)O3)=O)C2)ccc2nsnc2c1 c1(C(N(C2CN(C(C3(C)ON=C(C(C)C)C3)=O)C2)C)=O)cc2c(=O)[nH]ccn2n1 N1(C(c2c(F)ccc(NC(=O)OC)c2)=O)CC(C2CCCN(C(C)=O)C2)C1 C#CCC(CC(F)F)C(=O)N(CC(=O)NC)CC.C1(CN)CCN1CC C1(CNC(c2cn(CC)nc2)=O)CC(NC(=O)Cc2ccc(Cl)s2)C1(C)C Cc1c(Cl)c(C(=O)NC2CN(C(=O)CC3CCC=CCC3)CC2C)nn1C C1(NC(C(C)CN(C)C)=O)CC2(C1)CC2NC(=O)CNC(c1cscn1)=O Cc1cc(C)c(C(=O)NC2CCC3(C2)CN(C(c2cccc(Br)c2)=O)C3)cc1C C(=O)(C(C)(C)C(C)(C)O)N1CCC(OC)(CNC(=O)CCc2cnn[nH]2)C1 C(C(C(=O)N(C(C)C(=O)NCC1CCOC1C)C)OC)OC N1(C(C2C(C)CCOC2)=O)CCC(CC(=O)NCC2(CC(N)=O)CC2)C1(C)C Cc1nc2n(n1)CCCC2NC(=O)C(C1CC(F)(F)C1)N C1(NC(C2CCN(CC)CC2)=O)CC2(C1)CC(CNC(c1csnc1Cl)=O)C2 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC2(N(C(C=CS(C)=O)=O)CCC2)C1 c1(OCCOC)cccc(CCC(=O)NC2CC(F)(CNC(=O)C3CC3)C2)c1 c1(OC)cc(OC)cc(CC(=O)NC(CNC(C2CCC(C)O2)=O)CO)c1 c1(C(=O)NCC2CC(C)N(c3ccnc(C4CC4)n3)C2)noc2cc(Cl)ccc12 N1(C(C(C)NC(CC)(C)C)=O)CCCCC(C(=O)N(C)Cc2cnn(C)c2)C1 c1(CC)nc(C)ccc1C(=O)NC(CO)C(C)NC(=O)CC1(O)CCCOC1 C(=O)(CCCC(=O)NCC1(F)CCN(C(=O)C(F)n2ccnc2)C1)N(C)C c1(C(=O)NCCC2(O)CCN(C(CCS(C)=O)=O)C2)cc(Cl)c2[nH]c(O)nc2c1 N1(C(C=Cc2n(CC)ccn2)=O)CC(NC(=O)COC)CC(C)C1 N1(C(CC(C)C)=O)CCCOC(CCNC(c2cnnn2C)=O)C1 CCCCC(CC)CC(=O)NCC(C)(C)OCC(=O)N(CCc1ncon1)CC CCC(F)(F)C(C)(C)C(=O)NCC1CN(C(=O)CCOC(C)C)CCO1 CC(O)C(F)(F)C(=O)N1CCCC(CCC(=O)N(C2CCCC2C)C)C1 C1(C(=O)NCCCC=CC)CN(C(c2c[nH]cc2C)=O)CC1C1CC1 c1(CC)nc(-c2cccc(O)n2)n(C(C2(C)CC2)C)n1 C1(CCOC)(NC(C2CCCCC2O)=O)CCN(C(=O)CCCCN(C)C)C1 c1(NC(=O)NC(c2nc(C3CCCCC3)no2)C)cc(Cl)c(Cl)cc1Cl c1(C(=O)NCCNC(C(C)C)=O)n[nH]c2c1CN(C(=O)C=CC1CCOCC1)C2 C1(NC(=O)Cn2cncn2)CCC2(CCCN(C(=O)Cn3cccnc3=O)C2)C1 c1(OC)cnc(Cl)cc1C(N1CCC(CO)(NC(c2[nH]cc3c2CCC3)=O)C1)=O CN1CCC(C(=O)NCC2(C(=O)NCC3CCN(CC(F)(F)F)C3)CC2)C1 c1(-c2c(CNC)cccc2F)cccc2[nH]nc(C(=O)NCc3ccccn3)c12 N1(C(c2cc(C)nn2C(F)F)=O)CCCC2(CCN(C(C3(C)CC(C)C3)=O)C2)C1 C1(NC(c2ccc(COC)[nH]2)=O)CCN(c2nc(Cl)ncc2C)CC1(C)C CCCCS(=O)(=O)CC(=O)N1CCCC1CCNC(C1COCC(C)(C)O1)=O C1(NC(Cc2cc(C)nn2C)=O)CC2C1CCN2C(c1ccoc1)=O c1(N2CCC(O)(CN)CC2)ccc([N+](=O)[O-])nn1.c1(OC)cccc(OC(N)=O)c1 N1(C(C2(CC)CN(C(=O)C(F)OC(F)(F)F)C2)=O)CCN(C)CC1C C12(C(=O)NC(C=C)CO)CCCC1CN(C(c1cc(O)ncc1F)=O)C2 c1(C(=O)NCC2(OCC)CN(C(=O)CSc3n[nH]c(=N)s3)C2)c(Cl)ccnc1C C(=O)(CC(C)(C)CNc1ccc(C#N)cn1)OCC1(OCC)CCOC1 c1(CN(C(=O)CC2(CC(=O)O)CC2)C(c2ccco2)=O)ncc(-c2cn(CC)nn2)o1 C1(C(=O)NCC(N2CCCC2)C)CN(C(=O)CC(=O)NC2CC2)CC(C)(C)O1 Cn1nnc2c1CCC(C(=O)NC1(C)CCN(C(c3nc(Cl)cs3)=O)C1)C2 N1(C(C(CC=C)C)=O)CCN(C(c2ccncc2Cl)=O)C2CC12 C1(C(N2C3C(NC(c4cccc(C)c4)=O)C(CC3)C2)=O)CCCC1P(C)(C)=O N1(C(c2ccccc2CO)=O)CC(CO)C2(C1)CN(C(C1CCCO1)=O)C2 c1(-c2n(CCCC)nc(CNCC)n2)ccc(C=O)cc1C.C1(CS)CC2CCC1C2.CCl.OC C1(CC)(NC(C2COC2)=O)CCN(C(C2CCN(C)C(=O)C2)=O)CC1 CC(C)CC(C)(CNC(C1(C2CC2)CC1)=O)NC(=O)C1=CCSC1 c1(N(C)Cc2c(CC)cccc2)nc(NC(C)C(C)CO)c2ncsc2n1 c1(CSCC(=O)NCC(CCC)NC(=O)CSCCN(C)C)c(C)noc1C c1(OCCC(=O)NCC23N(C(CCC)=O)CC(C2)C3)cccc2ccccc12 C1(O)(CCNC(CC(=C)C)=O)CCCN(C(c2c[nH]nc2C2CCCNC2)=O)C1 n1(CCN)nc(C(F)(F)F)cc1CO.C1(NC(C2(n3cccn3)CC2)=O)CC(CCF)C1 C(=O)(C(C)CC=Cc1cccs1)NC1(C#C)CCC1 N1(C(C2N(C(c3c(C)snc3)=O)CCSC2)=O)Cc2ncsc2C1 CC(N=c1nc2scnc2c(N2CCC(OCCO)CC2)[nH]1)C1CC2(CCC2)C1 CC1CCN(C(C2SCCCS2)=O)C1CNC(c1ccc(CO)s1)=O C(CCCCCNC(=O)Cc1cccc(C(F)(F)F)n1)NC(COCCCC)=O C1(NC(c2n(CC)nnn2)c2noc(C)n2)CCC2CC1CO2 CC1OCCC1(C)C(=O)NCC(C)(C)NCCNC(c1cc(CCN)ncn1)=O c1(C(=O)NC(CNC(c2c(C)c[nH]n2)=O)C2CCC2)cccc(F)c1N C12(COC(c3cc(C(C)(C)F)ncn3)=O)CC(C)(C1)C(CN)O2 C(C)(C(C)(C)NC(=O)Cn1nnnc1C)NC(CC1(OCC)CCC1)=O CCC(CC(=O)NC1CC(NC(=O)CC(C)C(=O)OC(C)(C)C)C1)C(=O)OC c1(C(=O)NCC2(F)CC(COC)C2)cncc(-c2ccc(Cl)cc2)c1 CC(O)(CC(=O)NCC(F)(F)Cn1cc(C2CC2)nn1)C1CC1.C1(C)CCCC2CC12 C(CN=c1[nH]nc(COC)s1)N(C(c1cnoc1C)=O)CC N1(C(C(CC)OCC)=O)CC2CN(C(=O)C=C(C)C(F)F)CC2(C)C1 O=C(CCCCC1CCC1)NCC1CC(F)C1.C12CCN1C2 c1(C(=O)NCCC2N(C(CC3(C#N)CC3)=O)CCSC2)cccc2nonc12 C1(NC(c2cn(CC=C)nn2)=O)CC(C(=O)NCCC2C=CCC2)CC1O Cc1c(N)ccc(C(=O)NCC2CCN2C(c2c[nH]nc2-c2ccco2)=O)c1F c1(OC)cc(NC(C)CNC(=O)Cn2cnc(C(N)=O)n2)nc(OC)n1 C1(NC(c2n(CCC)ncc2)=O)CCN(C(=O)C=CC2COC(C)(C)O2)C1(C)C C(=O)(C(CNCc1cn(CC(C)(C)C)nn1)CC(C)C)NC.c12c(C)nnn1C2 C(c1cccc(F)c1Cl)=CC(=O)NCC(C)CNC(C1CCO1)=O CC1CCC2(CCN(C(=O)C(=O)NCc3nccnc3-c3ccsc3)C2)C1 CC1(C(=O)NC2CC(C(=O)NCC3(Cl)CC3(F)F)CC2O)CCCOC1 c1(C(=O)NC2CN(C(C(C=CC)O)=O)CC2O)nc(C)ccc1C CC(C)CCOCC(=O)NCCSC1CC(OCCOCCCC2CCC2)C1 C1(NC(C2(CCOC)CC2)=O)CCN(C(C2CCCCC2C)=O)C(C)C1 C1(Nc2cc(CCC)ncn2)C2CCC(C2)C1CNC(C(=O)OC)=O C1(C(=O)NCC2C(OC)CC2)CCOC1CNC(=O)CCOC1CC1 Cc1ncc(C(=O)NCC(C2CC2)NC(=O)C(C2CCCO2)C2CC2)s1 Cc1nc(O)sc1C(=O)NC(C1CCCN1C(c1ccc(C2CCC2)nc1)=O)C c1(C(=O)OCc2ccc(C)nn2)c(-n2cccc2)sc2c1CCC2 N1(C(C(C)C2CCOC2)=O)CCC(O)C(CO)C1.C(C=O)NC1CC1 N1(C(C2CCCN2C2CC2)=O)CC(O)(CCNC(=O)CCCc2cnccn2)C1 c1(C(=O)NC2CC(O)CN(C(c3cnn[nH]3)=O)C2)ccc([N+](=O)[O-])cc1 C1(CNC(C(C)CO)=O)CCC2CN(c3cc(CC4CC4)ncn3)CCC2C1 C1(C(N(CCOCCCNC(C(COC)O)=O)C)=O)CC2(C)CC1CO2 O=S(=O)(c1ccc(Br)cc1Cl)N1CC2(CCCN(c3ncccn3)C2)C1 N1(C(C(C2CN(C(CCCC(C)C)=O)C2)O)=O)CC2CCC1C(O)C2O CCCCCC(O)CNC(c1ccc(CNC(C2CCC(C)O2)=O)s1)=O c1(C(=O)NC(CNC(C2CN(C(N)=O)C2)=O)C2CC2)cc2c(nn1)CCC2 N1(C(CC)=O)CCC(C(=O)NCCCN(C)C(c2ccc(C(C)C)s2)=O)C1 N1(C(c2cc(C#C)c(C)cc2)=O)CCC2(CCN(C(=O)CC(CC)CC)C2)C1 N1(C(c2cn(SCC)nn2)=O)CCC2CCN(C(c3cn4c(n3)SCC4)=O)CC12 CCC(CC)C(C(=O)NC(C1CCOC1)CNC(=O)C=C(C)C1CC1)OC N1(C(C2(CCC)CCC2)=O)CCC(C2(C)CC2)C1.C12CC1CC(=O)NC2 c1(C(=O)Nc2ncc(NC(C3(COC)CCC3)=O)nc2)ccc(Br)c([N+](=O)[O-])c1 C(=O)(C#CC1CCCO1)NC1C(CN(C(=O)Cc2cccs2)C)CCC1 C(=O)(C#CC(C)(C)O)NCC(CNC(c1cc(CC)n(C)n1)=O)(C)OC c1(C(N(C2CC2)CC2CCN(C(CN(C)CC)=O)C2)=O)ccccc1SC c1(CN(C)C(=O)NCc2[nH][nH]c(=N)c2Br)ccc(Cl)c(Br)c1 Cc1cccc(C(F)(F)C(=O)NC(CNC(=O)C(C#N)C2CC2)C2CC2)n1 C1(CNC(C2(CCNC(C=CC(CC)=CC)=O)CC2)=O)CCC(C(C)C)CC1 CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1CC(CNC(c2cc(N)cc(F)c2)=O)C1 N1(C(CCOC(C)=O)=O)CCc2c(c(CNC(C3CCC(C)C3)=O)nn2C)C1 C=CCC(CNC(=O)Cc1ncn(C)c1C)C(=O)NC(C=C)C1CC1 c1(CCC(=O)NCC(C(C)C)NC(=O)CN(S(C)(=O)=O)C)c(F)cccc1Cl C1(CNC(=O)Nc2cccc(C)c2)CCN(C(=O)C(O)C2CCCC2)C12CCC2 N1(C(c2cccc(Br)c2)C(=O)NCCCOC)C2CCC1C(C)C(O)C2 c1(C(C(=O)CCC2CC2(Cl)Cl)=O)[nH]nnc1C(=O)NC.C(CN)(C(C)C)N N1(C(Cc2n(C)nnc2)=O)CC(NC(c2ccccn2)=O)CC12CCCOC2 Cc1nc(CO)sc1C(=O)NCC1CC(O)CN1C(=O)C(C)n1cnnn1 Cc1ccc(Cl)c(OCC(=O)N(C(C)C(c2c(F)cccc2F)O)CCO)c1 C(=O)(C(CC(C)C)NC(=O)C(C)COC)N(C(CC)CO)C c1(C(=O)NCC(C)(C2CCC2)NC(c2cc(C)oc2C)=O)cn2c(n1)CCC2 C1(CNC(CC(C=C)CC)=O)C(C2CC2)CCN1C(c1cc(C)c(F)c(C)c1)=O N1(C(=O)NC(c2ccncc2)(C)C)CCOCC(C(=O)N)C1.c1(CC#N)ccccc1 C(=O)(CC(C(F)F)N(C)C)NC(c1cccnc1F)C.C12(CCC1)CC(=O)N2 C1(CC)(NC(=O)CC2CCCC(=O)N2)CCN(C(c2cc(F)cnc2O)=O)CC1 c1(C(=O)NCC(C)(C2CC2)NC(C2CC2F)=O)[nH]nnc1C1CCC1 c1(C(C#C)(C)NC(C2CCC2CC(=O)O)=O)ccccc1 c1(OC)cccc(C(=O)NC2COCC2CNC(c2ccnnc2O)=O)n1 CN1CCC2(CCN2C(=O)CC2CCCC2NC(=O)C=Cc2cocn2)C1 CCC(CC)(CCC(=O)N1CC(O)CC1CNC(=O)Cn1ccc(C)n1)[N+](=O)[O-] C(=O)(C(C)(O)C(C)O)NC1CCN(c2cccc(C)c2)CC1 c1(C(N2C(COC)CN(S(=O)(=O)CC3CCC3)CC2)=O)ccc2nc(Cl)sc2c1 C(C(C(=O)NCCn1ncccc1=O)C(C)C)NC(C(C)=CC=C)=O C1(O)(C(C)NC(c2ccc(C(C)C)s2)=O)CCN(C(C2CC(C)CO2)=O)CC1 CCCCS(=O)(=O)NCC(=O)NC1COCC1NC(C12CC(CN1C1CC1)C2)=O C1(NC(=O)CCc2nncnc2O)CN(C(c2cc(Cl)no2)=O)CC12CCOCC2 c1(NC(CC(CNC(c2[nH]ccc(=O)c2C)=O)OC)=O)cc(F)c(C)cc1F C(=O)(C(=O)C(C)CC)N1C(C)(C(N(CC#C)CCOC)=O)C=CC1 c1(C(N2C(C)CC(NC(CCOCC#C)=O)C2)=O)nccc2ccccc12 c1(C(=O)NC2C(CNC(c3cc(C)sc3C)=O)CC2)c(O)nc(=O)n2c1CCC2 N1(C(C2C(C)=C2)=O)CCC(NC(=O)CCc2cccc(F)c2Cl)C(CO)CC1 C1(C(N(C)CC2(CN(C)C)CC2)=O)(CO)CCCCC1.N12CC3CC3(C1)C2=O N1(C(C2CC(=O)C2)=O)CCOC(CNC(C2(c3cccs3)CCCCC2)=O)C1 C1(NC(C(c2c(OC)cccc2)C)=O)CN(C(c2ccnnc2)=O)CC1C#N N1(C(c2cnc(C)n2C)C(=O)NCC2CCCC2)CC(C)(C)OC2COCC12 n1(CC)cc(Br)c(C(=O)NCC2CCN(C(C3CC3(C)Br)=O)CC2)n1 CCS(=O)(=O)CCC(N)C(=O)N(C)Cc1ccc(Cl)c(C(F)(F)F)c1 Cc1c2ccc(NC(C3(Cc4ccncc4Br)CCC3)=O)cc2nn1C N1(C(=O)CNC(=O)C(F)(F)F)CCN(C(C2OCCO2)=O)C2CCCCC12 O=C1CN(C(=O)C(=O)N(Cc2ccc(Br)cc2)Cc2cccnc2)CCN1 C1(C(=O)NCc2nc(C)c(C)[nH]2)C2CCC(C2)C1NC(=O)C1=CCCC1C C1(CNC(C2C(CC)C2)=O)CN(C(=O)C(C)Oc2ccccc2F)CCN1C Cc1c(C(=O)NC2CN(C(c3ccnc(C(F)(F)F)n3)=O)C2)cccc1O c1(C(=O)NCc2cn(CCN(C)C)nn2)cc(-c2ccco2)nnc1O C(N=c1[nH]ccnc1Br)c1cncc(C(=O)NC2CC2)c1 c1(C(C)C)ccc(C(N2CC(O)CC2CNC(C2(C)COC(=O)C2)=O)=O)nc1 c1(C(CCC(=O)N2CC(NC(C=C3CCC(C)C3)=O)C2)=O)coc2c(Cl)cccc12 c1(C(=O)NC2CN(C(c3c(CC)nccc3)=O)CC2C)ccn(C)c(=O)c1 c1(C(=O)NC2CC(C)(NC(Cc3scc(C)c3)=O)C2)c(N)cc(Cl)nc1Cl CCC(CNC(=O)C(CC(C)C)ONC(C1CCCSC1C)=O)(CC)CO C1(NC(CCC(C)SC)=O)CN(c2nc3ccccc3s2)CCC12CCOCC2 c1(C(C)C)nn(C)cc1C(=O)NCC1(C)CCN(C(C2CCCC2(F)F)=O)C1 c1(C(=O)NC(C(C)C)CNC(=O)CCOC2COC2)cccc(N2CCCC2)c1 N#Cc1cc(NC(c2cncc(-c3ccsc3C#N)n2)=O)cnc1Cl C1(NC(=O)CC2C=CCCC2)CC=C(C(=O)N2CC(CO)(CO)C2)C1 CN1CCCCC1CCNCCCNC(c1nc(C2CC2)cs1)=O c1(SC(C)CN(C(=O)CC2(C)CCCC2)C)ccccc1Cl.C1(C(=O)N)CC(C)(C)O1 N1(C(C2(CC#C)CC2)=O)CCC(CNC(=O)CC=CI)C1 Cc1cc(F)cc(C(=O)NCC2CCN(C(C3(C)CC3C)=O)CC2O)c1N C1(C(=O)NC2CC(C)(C)C2)CCN(C(c2cnc(O)o2)=O)CCO1 C(=O)(C(C)(C)S(C)(=O)=O)OCC(C)(C)N(C(COC)=O)C C1(CC(=O)N(CC(CC)NC(c2cc(C(N)=O)cs2)=O)C)CCC2CC1C2(C)C N1(C(=O)NCC(C)CC2(C)OCCO2)CCc2cc(Br)c(F)cc2C1 c1(OCC)cc(NC(C2CC2CC2CCC2)=O)ccc1NC(n1cc(Br)cn1)=O C1(CCNC(=O)CCCc2ccccn2)CCCN(c2nnc(O)s2)C1 C=C1CC2CCC(C1)N2C(=O)CCC(C)(C)NC(=O)CS(C)(=O)=O C(=O)(C(C(C)C)c1cccnc1)N(C1CCCCC1)CCNC(C1(SC)CC1)=O c1(C(C)C(=O)NC(C)CCCNC(=O)C(F)n2ccnc2)cccc(F)c1 CC1C(NC(c2ccsc2Br)=O)CCCN1c1cncc(C(F)(F)F)n1 CCC(C)C(=O)C(=O)NC(Cc1cn[nH]c1)C(=O)Nc1ccsc1C C(CC(C(C)C)N1CCOCC1)NC1(SC)CCCCC1 N1(C(C2(C#N)CCC2)=O)C2CCN(C(c3ccc(-c4cccnc4)cn3)=O)CC12 C1(NC(C2CCCOCC2)C)CCCc2ccc(Br)cc2C1 c1(C(N2C(C)CC(CNC(=O)C(F)=CC3CC3)C2)=O)cnc2cnc(Cl)cc2c1 C1(NC(c2c(C)c[nH]n2)=O)CCN(C(=O)C=Cc2nnn(C)n2)C1C CC1=NOC(C(=O)NCC(C)(F)CNC(=O)Cn2ncc(Br)n2)C1 N1(C(c2ccc(C)c(F)c2)=O)CCC2(CCCN2C(=O)C(C)N2CC(C)C2)C1 N1(C(Cc2c(C)cco2)=O)CCn2ncc(S(C)(=O)=NC(=O)CC(C)O)c2C1 c1(NCC(N(CC)OC)=O)nc2ccccc2nc1NC(CSC)C1CC1 C1(NC(C(C#C)(C)C)=O)CC2(CCC(CNC(C3CCN(C)C3=O)=O)OC2)C1 CCCCCC(O)CC(=O)NCC(C)N(C)C(c1cncc(C(=O)OC)c1C)=O N1(C(C)C)CCCC(C(=O)NCCC(C)CCNCC=Cc2ccncc2)C1 N1(C(C(C)OCOC)=O)CCCCC(NC(c2cncc(C)c2)=O)C1 c1(OC)ccnc(C(=O)NC2CC(CNC(c3n[nH]c4c3CCC4)=O)C2)c1O c1(OC)ccc(C(=O)N(C)Cc2cn(-c3ccc(CNC(C)=O)cc3)nn2)cc1 Nc1cccnc1C(=O)NC(CCF)C(=O)NCCC(Cl)Cl c1(CNC(CC2C(NC(COC)=O)COC2)=O)nc(C)c(C)o1 C1(C)(CNC(CC2CC(OCC)C2)=O)CCN(C(=O)Cc2ccccc2O)C1 C1(NC(CC)=O)CS(=O)(=O)CC1N=c1[nH]nc(-c2ccccc2)s1 N1(C(CCc2n(CC)ccn2)=O)C2CCC1CC(NC(c1nc(C)sc1C)=O)C2 CC#CCC(C(=O)N(C)Cc1cncn1C)NC(c1nccs1)=O S(=O)(=O)(c1ccsc1C(=O)Nc1ccc(N(C)C)cc1)NCCN(C)C c1(OC)cccnc1CNC(=O)C=CC(C)NC(=O)CC1CC(CC)=NO1 c1(C(=O)NC2CCN(C(C(CCC)OC)=O)C2C)oc2ccccc2c1CC C1(C#N)(C(N(CC(C)N(C)C(C2CCS(=O)(=O)N2)=O)C)=O)CC=CC1 C1(COC)(CNC(=O)Cn2cc(C(C)O)nn2)CCN(C(=O)CCCC2CC2)C1 c1(C(=O)NCC=C(C(=O)NCc2cn(CC=C)nn2)C)cncc(C)n1 c1(-c2nc(CSC)nn2C2CCOC2)cc(F)cc(Br)c1F C1(NC(C2C(C)(C)CC2)=O)CC(F)CN(C(=O)CSc2ccccn2)C1 N1(C(C(N2CCCC(C)C2)=O)=O)CC2CC(O)C1C2NC(C1CCCN1C(N)=O)=O C=CC(CC)CC(=O)N1CCN(C(=O)CN2CSCC2=O)C(CC(F)(F)F)C1 c1(NC(C2(C)CCCN2c2cnc(C#N)cn2)=O)cccc([N+](=O)[O-])c1 N1(S(CC#N)(=O)=O)CCCC12CCCN(C(=O)C1CCCc3ccccc31)C2 C1(O)(CNC(C(C)(CO)NC(=O)OC)=O)CCCN(C(=O)C(F)F)C1 N1(c2cc(C)nc(N3CCCOCC3)n2)CCCC2(C1)NC(=O)NC2=O.CO c1(NC(=O)NCC2N(C(C3(C=C)CCC3)=O)CC2)cc(C)c(Cl)cc1OC C1(C(=O)NCC2CCCN(C(C)C)C2)C(c2ccccc2)C2CC1C(O)C2O C(C1=NOC2CN(C(c3coc(Cl)c3)=O)CC12)NC(=O)CSc1ccc(O)cc1 c1(C(N2CCC(C)(O)C2)C)ccc(-c2cnn(CCN3CCCCC3)c2)nc1 c1(C(C(=O)NCCC(C)NC(C2CC2C)=O)(C)O)ccc(Cl)cc1 C(CCCOC)(C(=O)N1CCC(O)(C(F)F)C1)NC(CCC)=O N1(C(C(c2ccc(OC)nc2)(F)F)=O)CCC(NC(c2cc(C)sn2)=O)C(O)C1 CC1CC(C(N2CCN(S(=O)(=O)Cc3ccccc3)CC2)=O)N(CC2CC2)C1 c1(CNC(C(C2(O)CCC2)NC(c2cc(OCC)n[nH]2)=O)=O)nccnc1C C(=O)(C1=CCC2(COC2)OC1)NC(CNC(CN(C(C)=O)C)=O)CCOC S(=O)(=O)(C(F)(F)F)NCC(=O)NC1CCC1NC(c1ccc(CO)cc1)=O C12(NC(c3c(C)nsc3)=O)CCCC1CN(C(=O)Cc1c[nH]c3ccncc13)C2 N1(C(CCCc2nc(C)sc2)=O)CCCC(CCNC(c2cnc(Cl)s2)=O)CC1 c1(CNC(=O)C=CCBr)ccc(CNC(c2coc(Cl)n2)=O)cc1 c1(C(=O)NC2C(C)(C)CN(C(C3CSC3)=O)C2)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(c2cc(C)nc(O)n2)=O)CCC2(CC1)CC2NC(=O)CN1CC(=O)NC1=O C(C(C(=O)NCCC1CCC(=O)N1)C(C)C)NC(C1(C#C)CC1)=O c1(OC)ccc(CNC23CC(C(=O)NCCCc4ccccc4)(C2)C3)cc1Br CN1CCN(C(CC=CCC2(C)CC(C(=O)OC)C2)=O)C(C(N2CCCC2)=O)C1 Cc1cc(CNC(=O)C(CN(C)C)NC(=O)C=CC(F)(F)F)no1 c1(NC(C2=CC=C2Cl)=O)cc(-c2ccco2)c(-c2cccn2C2COC2)cn1 N1(C(c2cc(CO)on2)=O)CCCN(C(=O)C(c2ccc(Br)cc2)O)CC1 c1(C(=O)Nc2cccc(OC3CC3)c2)cc2ccc(Br)cc2nn1 CC(C)CC(CNC(c1ncoc1C(C)C)=O)C(=O)NCC(C)(C)C1CC1 c1(CN(Cc2ccc(OC)cc2)CC2(C)C3COCC23)c(C)cc(OC)cc1C c1(C(=O)NCC23CC2CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C3)cnc2ncccn12 c1(C(=O)NCC2(CCNC(C(C(C)O)N(C)C)=O)CC2)ncc(Cl)c(N)c1Cl CC1(O)CON(C(=O)C2CC3CN(C(c4cnsn4)=O)CC3C2)C1 c1(-c2nc(C(C3CC3)OC)nn2C(C)C)c(F)cc(F)cc1F CC(O)C(C)(C)CNC(=O)NCCn1cnccc1=O N1(c2c(Br)cnc(OC)n2)C2CCC1CN(C(=O)Cc1ccc(F)cc1C)CC2 c1(C(N2CCCC(CC(=O)NCC(N3CCCC3)C)C2)=O)cc2cccn2cn1 C1(C(=O)NCCNC(=O)C=CCO)CCCN(C(=O)C=CC2CCCCC2)C1 C(=O)(C1=CCCOCC1)N1CCC(C(=O)NOCC2CCCO2)(CC#C)C1 C1(C(=O)NC2(C(=O)NC3CCC(CO)CC3)CC(O)C2)CC1C1CCOCC1 C1(CCC)CN(C(c2ccc(Cl)c(OCC)c2)=O)CCN1C(=O)C=C1CCC1 N1(C(C(CCOC)C)=O)CCC(NC(=O)CC(=O)NC2CC2)C12CC2 Cc1ccncc1C(=O)NC1CCC(C(=O)NCC2(C)CC(C)(C)C2)C1 c1(CC)cc(C)ccc1C(=O)NC(C)C(CO)NC(C1CC(C)(C)C1)=O CC1COC(CC(=O)N(C)CC2(CNC(c3ccc(-c4ccco4)[nH]3)=O)CC2)C1 CC1(C)CC(NC(=O)C(C)(Cl)Cl)CCN(C(C2(C(F)(F)F)CC(O)C2)=O)C1 c1(C(N2CCC(C(C)C(=O)NCCOC3CC3)C2)=O)csc(C#N)c1 C1(C(N2CCC(N(C(c3n[nH]c(C)c3Cl)=O)C)CC2)=O)CCC12CCCO2 C(=O)(C(CN(C)C)C(C)C)N(C)CC1(CC)CC1.C12CCCCC1C(=O)N2C N1(C(C(C)C(F)F)=O)C2CCC1CN(C(=O)CN(C)C(N)=O)CC2 C1(C(=O)NCCN(C(c2cccn2C(C)C)=O)CC)CC2CCC(C1)N2C C1(C(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)OCCOC1(C)C C#Cc1ccc(C(=O)NC2CC(C(=O)NCC34CCC(CC3)O4)C2(C)C)cc1C CCC(O)C(C)(C)C(=O)NCC1CC1NC(c1csc(Cl)c1)=O Cc1c(Br)ccc(C(=O)NC2C3CN(C(c4c(C)cc(Br)cc4C)=O)CC23)c1F C1(OC)CC(CCNC(=O)CCc2ccnn2C)N(C(=O)C=CC2CCOC2)C1 N1(C(=O)COC2CC2)CCCC(CC2CCN(C(=O)CCOCC3CCCO3)C2)C1 c1(C(N2CC(CCC)N(C(=O)CCCCOC)CC2)=O)cc(F)cc(N)c1F C1(OC)CCCCC1C(N1CCCC1)=O.C12CC(C1)C(=O)NCC1CC1C(=O)N2 C1(OC)CN(C(C2CCC=CCC2)=O)CC1NC(c1cnc(C)n1C(F)F)=O C12(C(=O)N(CC(=O)NC(c3cncc(Br)c3)=O)CCO)CCC(C3CC3)(CC1)CC2 N1(C(C=C2CCN(C)CC2)=O)CCC(CNC(=O)Cn2cccn2)C(F)(F)CC1 N1(C(c2c(C)nc(C(F)(F)F)o2)=O)CCN(C(=O)C(O)P(C)(C)=O)CC1C1CC1 Cc1cccc(C(=O)NC(C)C(=O)NC2C3CN(C(C4(Br)CC4)=O)CC23)c1 N1(C(CCC2CCN(C(=O)CN3C(=O)CCC3=O)C2)=O)CC2CCCCC12 c1(NCCC(=O)NCC(C)NC(c2cscc2F)=O)c(F)cccc1F C(=O)(C(C)(C)CF)NCCCN(C(CCc1ncn(C)c1)=O)C1CC1 CCCCCCCCOCC(=O)NC(CN(C(=O)C=CCOC)C)CC c1(C2CC(C(=O)NC(CCNC(COC)=O)C)C2)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(CNC(CCCOCC=C)=O)CO)nn(C)c(Br)c1C c1(C(CC(=O)NC(CC(C)NC(c2ccncn2)=O)C)C)ccc(Cl)cc1 C1(C(=O)NC(c2c(C)n(-c3ccc(F)cc3)nc2)C)CC(F)(F)CCC1(C)C N1(C(C2CCOC2)=O)CCC2CC(NC(C3(c4ccoc4)CC3)=O)CCC2C1 c1(CC(=O)NC2(CNC(Cc3c(C)ocn3)=O)CCCC2)cnn2ccccc12 C#Cc1cccc(CC(N2CC(C(=O)NC(C)COCC)C3(CC3)C2)=O)c1 C(=O)(C1=CCCN(C(C2(n3[nH]cnc3=N)CC2)=O)C1)NCC(CC(C)O)C NS(=O)(=O)c1n[nH]cc1C(=O)NC1C2CN(C(=O)Cc3csc(S)n3)CC12 c1(C(=O)NC2CCN(c3nnc(C4CC4)s3)CC2)cccc2cnsc12 c1(-c2cn(C3CCCN(C(c4cc(COC)oc4C)=O)C3)nn2)c(F)cccc1F C(N=c1cc(C)nc(C(C)C)[nH]1)C1(O)CN(C(C(CCC)S(N)(=O)=O)=O)C1 C(=O)(C1CCc2cccnc21)N1CC2(C(NC(CCCC(N)=O)=O)CC2)C1 C1(CNC(CCOC(C)=O)=O)COC(C)(C)CN1C(=O)Cc1cnc(C)s1 N1(C(C2N(C(c3cc(COC)on3)=O)CC(C)C2)=O)CCCC(C)C1CO CCCCCCCCC(F)C(=O)NCCC(C)NC(=O)Cn1ccc(C(F)F)n1 C(=O)(C1=CCCCCC1)NCC1(C)CCCN(C(C2COC3(CO)CC2C3)=O)C1 Cn1cc(C(N2CCC(O)(CNC(=O)Cc3cnc[nH]3)C2)=O)c(Br)n1 c1(C(=O)NC2C(NC(c3c(C)ccc(Br)c3)=O)C2)cc(C)c(C)c(F)c1 Cn1c(=O)c(CNCC2C3CNC2C3)cc2ccccc12 C1(CC(=O)NCc2ccn(C)n2)CCCCC1NC(C12CCN(CC1)C2)=O C(=O)(C1CCCn2cncc21)N1C(CNC(c2oc(C)c(Br)c2)=O)CC1 c1(N(C)C)ccc(C(=O)NC2CN(C(=O)CC3COCCOC3)CC2O)c(F)c1 CCCN=C(NCCC(=O)OC)NC1CC(OC)C12CCC2 N1(C(CC2(OCC)CC2)=O)CCCC(CNC(=O)C(C)(C)OCOC)C1.C(=O)O c1(COC)ccccc1CNC(=O)N(C1CCC1O)C N1(C(c2ccn(CCN)c2)=O)CC2CC2C1.n1(CCCN(C)C)cnc(C(=O)O)c1 c1(C(C(=O)NCCCCCC)N(C(C)(C)CO)C)ccc(Cl)c(F)c1 c1(C(=O)N(C2CCCCCC2O)C)ccc(S(C)(=O)=O)[nH]1 C12(C(=O)NCCOCCCNC(=O)CC3CC(C(F)F)C3)CCCCC1C2 Cc1cc(C(N2C(C(=O)NC3CCCC3)CCC2C2CC2)=O)cnn1 C1(C(N(CC#CC)CC#C)=O)CC=CCN1C(C1CCNC1=O)=O CCC(C(=O)OC)C(=O)NCC1=CCCN(C(C2C=C(C)CS2)=O)C1 C1(C(=O)NCC2(C(=O)NC(C3CCCCC3)C)CC=CC2)CCCC(=O)C1 C(CC(C)C(=O)OCC)NC(C(=O)NCc1cn(CCC)nn1)C1CC1 C1(NC(CCN(CC(C(C)C)C)C)=O)CN(C(=O)C=C(Cl)Cl)CC2CC12 C1(C(N2CCC(NC(c3c(OC)csc3)=O)CC2C)=O)CC2(CCOCC2)C1 C(CC(C)(C)C(=O)NCCCCCC(=O)NCc1cnc(C)cn1)SC C#Cc1cc(C(N2CCCCC2CNC(=O)COC)=O)ccc1C C1(C(=O)NC2CC(F)(COCC)C2)(NC(=O)CCc2ccccc2)CCCCC1 Cc1cnccc1C(=O)NC1CCN(CCOCCC(C)C)CC1 CC1OC2CCC1(CNC(=O)C(C1CCN(C(=O)C(C)(C)CO)C1)C)C2 C1(CC#C)(C(=O)NC2CCC2NC(=O)CCC2CCCO2)CCOC1 N1(CC(=O)NC2CC2C(c2ccco2)=O)CCN(c2ncco2)CC1 Cc1ncc2cc(C(=O)NCC(O)CNC(c3ncn(C(C)(C)C)n3)=O)ccn12 c1(C(N2CCCC(NC(COCC)=O)C(F)C2)=O)cnc2c(c1)C(=O)CCC2 Cc1ncc(C(N2CCC(CN(C(=O)CC3COC(=O)C3)C)C2)=O)cc1N Cc1cc(CC(=O)NCCC2CCCN2C(c2nccs2)=O)cc(F)c1 C(C)(CO)(C(=O)NC1(CC(=O)NCCC2(O)CCOC2)CC1)OC C(=O)(CCP(C)(C)=O)N1CCC(C2N3CCCC32)CC1.Cn1ncc2c1C(F)C2 c1(OC(C)(C)C)cc(=NC(=O)c2csc(-c3ncccn3)n2)[nH]o1 N1(C(CN(CCC)C)=O)CCC(NC(=O)C(C)(C)C2CCOC2)C(O)C1 Cc1coc(C(C)C)c1C(=O)NCC(C1CC1)N(C(=O)Cc1csc(=N)[nH]1)C N1(C(COCCOCC)=O)CCCC(C)C1CNC(C1CCOC(C)(C)C1)=O c1(CC)ccc(C(N2CCC(NC(c3n[nH]cc3C)=O)C(CO)C2)=O)cc1Cl N1(C(C(C)(C2CC2)OC)=O)CCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC1 CN1CCOC(C(N2CCOCC(NC(=O)CSc3ccccc3)C2)=O)C1=O N1(C(c2c(NC)cncc2)=O)CC(CC(=O)NC2(CO)CCSC2)C2(CC2)C1 CCC1=C(C(=O)N(C2CC2)CC2CCCN2C(C23COCC2C3)=O)CCCO1 N1(C(C=C(C)C(C)C)=O)CC(NC(c2c(C)oc(C)c2C)=O)CC12CCCC2 N1(C(C(C)C2CC2)=O)CCCC(C2CCCN(C(=O)Cc3ccnnc3O)C2)C1 C1(C(=O)NCCN(C(=O)CCn2cccc2)CC)CC(CCOC)C1 C1(C(N(CCN=[N+]=[N-])CC)=O)CN(C)CCN1C(c1ncn(C)c1C)=O N1(C(C(C2CC2)OC)=O)CCC2(CCCN2C(C2CCCC(C)CC2)=O)C1 c1(NC(N(CCN(C)C)Cc2ccncc2)=O)cc2ccccc2nc1C(F)F c1(OC)ccc(C(N2CC3CC2CC3NC(c2cnnn2C)=O)=O)c(OC)c1.COC c1(C(N(C)CC2CCN(C(COC)=O)C2)=O)cc2c(cc1N)CCCC2 C#CCC(C)(C(=O)N1CCC(C#C)C1)NC(=O)C(C)N(C)C(C)=O N1(C(C(CCN(C)C)NC(=O)C#CC2CC2)=O)CC2CCC(C1)C2O C1(C(=O)NCCC2CN(C(=O)C3=CCCS3)CC(C)O2)CCCN2CCCC12 Cc1ccc(F)cc1C(=O)NCCCCC1CN(C(C2CC2(C)C(F)(F)F)=O)C1 N1(C(C(C)Cc2ccccc2)=O)C2CCCC1CC(C(=O)NC1CCCCO1)C2 Cc1cc(C(=O)NCCN(C(c2cc(Br)n[nH]2)=O)C(C)C)nc(C(F)F)n1 c1(C(=O)NC(CN(C(c2n(C(C)C)ncc2)=O)C)C)c(Cl)cccc1Br C1(CC(=O)NCCN(C(C(CCCC)C(C)C)=O)C)CCc2ccccc2C1=O C1(C(N2CCN(CCCC)CC2)=O)CCCN1NC(=O)C(F)C1CCCC1 CC(C)C(C)(O)C(=O)NC1CCC(NC(c2ncc(F)cn2)=O)C1 CCC(C)C(C)C(=O)N1CCCC(Cn2cc(COCc3ncccc3F)nn2)C1 c1(OC)ccc(C(N2CCC(C(C)NC(C3(CO)CCOC3)=O)C2)=O)nc1 c1(C(=O)NCC(CNC(C2CCCO2)=O)C(F)(F)F)c[nH]c2cc(F)c(F)cc12 C1(NC(c2c(COC)cco2)=O)CCCN(C(c2cn(C)nc2C(C)C)=O)C1 N1(C(C(C)(O)C2CCC2)=O)CC2CCC2(CNC(=O)Cc2cccc(F)c2)C1 c1(SCC(=O)N(C)CCN(C)C(C2(C)CC2(F)Cl)=O)ccc([N+](=O)[O-])cc1 c1(C(c2nnnn2C2CC(F)(F)C2)NCCC(C)CO)ccccc1[N+](=O)[O-] N1(C(CC2(COC)CCCC2)=O)CC2CC2(NC(=O)C(C)NC(=O)C2CC2)C1 c1(C(=O)NCC(c2ccc(Cl)cc2)NC(=O)CC2CC2)cnc(O)c(F)c1 N1(C(=O)CC2CCC2)C(CNC(C23COCC2C3)=O)CC2CCCC12 C=Cn1nccc1C(=O)NCC1CC(F)CN1C(c1sc(CO)nc1C)=O c1(OC)cc(C(C2CC2)NC(CCOCCO)C(=O)OC)ncn1 C1(C(=O)NC2(CNC(CN(c3ccccc3)C)=O)CC2(C)C)CCCC(=O)N1 Cc1cnc(NCC2(C)CCOC2)c(S(=O)(=O)NC2CC=CCC2)c1 N1(C(C(OC)OC)=O)CC(O)(C2CCN(C(c3cnccn3)=O)CC2)C1 C(CN=C(NCC1CCC(C)C1)N(C)CC(C)(C)OCc1ccccc1)SC Cc1cnc(C(=O)NC(C)CCCNC(=O)CC2CCNC2=O)c(Br)c1 c1(C(N(c2nc(CN3CC(N)CC(O)C3)cs2)CC)=O)cc2c([nH]1)CCCC2 N1(C(COCCC=C)=O)CCC(c2cn(-c3ccccc3CC(=O)O)nn2)CC1 CC(C)C(O)C(C)C(=O)NC1(CNC(C2(C3CCCO3)CCCO2)=O)CC1 NS(=O)(=O)N1CCCCC1C(=O)NCC1(C)CNC(=O)O1 N1(C(C2N(C(=O)OC)CCC2)=O)CCN(C(C2CN(C)C2)=O)C(C(C)C)C1 C1(CNC(=O)C(O)Cc2ccc(Cl)cc2)CCN(CCC2CC2)CC1 N1(C(c2cn(CCC)nn2)=O)CCc2ccccc2C1CNC(=O)C(O)C1CC1 N1(C(C2C(C)C2)=O)CCCC2(CCCN2C(c2cncc3c2CCCC3)=O)C1 c1(-n2cc(C(CCC)NC(=O)CCSC(C)CC(C)C)nn2)nc(CC)sc1N Cc1nn(CC(F)(F)F)c(C)c1CC(=O)NC1CCNCC1C#N C1(CNC(CC=CC=C)=O)CN(C(=O)Cc2nnc(C)s2)CC12CC2 C1(C)(CNC(C2CCC(CC(C)C)CC2)=O)CN(C(=O)C=CC(N)=O)CCO1 c1(C(C)C)c(C(=O)NC2(C)CN(C(=O)C(C)Oc3ccc(F)nc3)C2)cnn1C C1(c2n(CC=C)nnn2)(NC(C)CCC=CCC)CCN(c2ccccc2)C1 C12(NC(=O)Cc3ccc(CO)cc3)CCCN(C(=O)CCC3(O)CCC3)CC1C2 C(CC(CC)C(=O)NCCOCCC(=O)NC(C)C1CC1)=CC N#Cc1ccc(F)cc1C(N1CC=CC1C(=O)NCCn1ccnn1)=O C(=O)(C(CCc1ccccc1)NC(=O)C(C(C)C)OC1CCCC1)OC CCC(CC(F)(F)F)C(=O)NC(COC)CNC(=O)C(C(CC)CC)OC C(=O)(C(CCCC)C(C)C)NC1(CC=C)CN(C(c2nc(C)ncc2Br)=O)C1 N1(C(CCC=CC(C)C)=O)CCC(OCCNC(C2CC2Cl)=O)CC1 Cc1nc(CO)sc1C(=O)NCCC(C)NC(=O)C(F)(F)c1cscn1 C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1CCC(NC(c2ccc(SC)o2)=O)(CF)C1 c1(C(N2CCN(C(C3C(OCC)C3)=O)C(C(C)C)C2)=O)nc2ccccn2c1F CC(C)(O)C(F)(F)C(=O)N1CC(C(N)=O)(CNC(C2(C)CC2(F)Cl)=O)C1 Cc1ccccc1OCC(=O)NC1CCCC(NC(=O)C(O)C2CCC2)C1 c1(SC)cc(NC(=O)C(C(C)(C)C)n2ccnn2)ccc1F Cc1cc(Cl)cc(C)c1C(=O)NCCC1COCCN1C(=O)CCS(N)(=O)=O c1(OC)ccc(F)c(Br)c1C(=O)NC1CC(O)CN(C(=O)C(F)=C(C)C)C1 C(CCCCCNC(C1CCS(=O)(=O)C1)=O)NC(=O)CCc1cnccn1 C1(NC(N2CCN(CCN3CCCC3)CC2)=O)CCCC12CCC2 C=CCC(F)(F)C(=O)NCC(C(=O)NCCOc1cccnc1)C(C)C C(CC(C(=O)N(C1CCSC1)C)NC(c1coc(C2CC2)n1)=O)=CC Cc1cc(C)c([N+](=O)[O-])cc1NC(C1CC1NC(=O)Nc1ccc(Cl)c(F)c1)=O C1(C(N2C(C)CCC(NC(=O)CCc3ccc[nH]3)C2)=O)CN2CCCC2CO1 N1(C(CNC(CNC(C)=O)=O)=O)CCN(C(c2c[nH]nc2F)=O)C(C(C)C)C1 C1(NC(=O)CN2CC3CC3C2)CN(C(=O)CN2CCC(O)CC2)C2(CCCC2)C1 c1(C(=O)NC(C(=O)N(CCn2cnnc2)CC)C2CC2)ccc(N)cn1 C1(CC(=O)N(C2CN(C(CNC(c3ccc(C)s3)=O)=O)C2)C)CCCCCC1 c1(C(CN(C(C#C)CO)C)O)ccc(Br)cc1 c1(CC(=O)NCC2C=CCN2C(C2CCCCC(=O)N2)=O)cccc2[nH]ncc12 CN1CCC(CC(=O)NC2(C(=O)NCC3(C)CC4CC4C3)CCCC2)C1=O N1(C(C(CC)(F)F)=O)CCC(NC(C2CCCC2C2CC2)=O)C2(CCC2)C1 C(=O)(CC(C)C(=O)c1ccccc1)N(CCCNC(=O)CSC(F)(F)F)CC N1(C(=O)OC(C)(C)C)CCN(CCO)C2(CCCCC2)CC1.CCCSC C1(CNC(CC2CC(=C)C2)=O)CCN(C(=O)CCCCC)CC1C c1(OC)ccc(C=CC(=O)NCC(C)(C)CNC(c2ccc(F)s2)=O)c(C)c1 c1(C(=O)NCC(C2CCOC2)NC(CC2(C)CCC2)=O)ccc[n+]([O-])c1 Cn1ccc2c1CN(C1CCN(C(=O)C(F)C3CCNC3)C1=O)CC2 c1(C(N2CC(CC)N(C(=O)CCS(C)=O)CC2)=O)c(OC)ccc(SC)c1OC c1(C(N2CCCC(NC(CC(C)OC)=O)C2)=O)cccc(C)c1C#N C1(CN(C(C(COC)O)=O)C)CCCCN1C(=O)C(C)O C(=O)(CCCC(=O)NC1CC(C)CN(C(C2(CS(C)(=O)=O)CCC2)=O)C1)OC C1(C(=O)NCC(=O)NCCC)CCCC1CNC(c1csnc1C)=O C1(NC(Cc2ncc(C)s2)=O)CN(C(c2cccc(C3(C)CC3)c2)=O)CC1C C#Cc1ccc(C(=O)NC2CCCC2CC(=O)NCc2nc(CC)no2)c(F)c1 C(=O)(C1=C(C2CC2C)N(CC2CCCO2)C(=O)NC1c1cccnc1I)OCC c1(N2CC=CC(NCCCNC(C(C)=C(CC)C)=O)C2)c([N+](=O)[O-])cnn1C N1(C(C(CC)C(=O)OC)=O)CCN(C(=O)C=C(C)c2ccc(F)cc2)CC(O)C1 C1(C)(CNC(C(c2cnn(C)c2)C)=O)CCN(C(=O)CCC(C)(C)C)CC1 c1(C(=O)NC(CC=C)CNC(c2cc(C(C)(C)O)on2)=O)cccc(C(=O)OC)n1 c1(CN=C(N(C)Cc2ccnn2C)NCc2ccco2)cccc2oc(=N)[nH]c12 Cc1ccc(C(=O)NC2CCN(C(=O)Cc3cn4ccsc4n3)CC2C)c(C)c1 c1(C(C(=O)NC(C2CCOC2)CNC(CN(C)CC)=O)(F)F)cc(F)ccc1F C1(CN2CC(=O)N(C(=O)OC)C2=O)CC(CC2CN(C)C2)C12CCCC2 C(C1CCCN1C(=O)C=CC(F)(F)F)=CC(=O)NC(c1cnn(CCF)c1)C c1(C(N2C(CNC(c3onc(C)c3C)=O)CC2)=O)ncc(Cl)c(N)c1Cl Cn1cc(CC(N2CC(C)(CCC(N3CCC(CO)C3)=O)C2)=O)cn1 CC1CC(O)CCN(C(C23CC(C)(CN2C(c2ccsc2)=O)C3)=O)C1 c1cc(CNCC2CC3(CCC3)C2)ccc1N1CCOCC1 Cc1nc(C2CC2)oc1C(=O)NC1CC(NC(C2CCCC2(F)F)=O)C1 c1(C(c2n(-c3ccc(OC)cc3)nnn2)NC(C2(C)CC2)C)c(F)cccc1Br c1(OC)ccc(NC(=O)CC2(C)CN(C(c3ccc(=O)n(C)c3)=O)C2)cc1F CC1CN(C(c2csc(CNC(C3CCCCO3)=O)c2)=O)CCC1(F)F c1(C(=O)NC2CC(NC(CCN3CCC(C)CC3)=O)C2)cccc2c1OCC2C C1(CCC)CCN(C(=O)C(c2ccoc2)NC(=O)C(C)OC(C)=O)CC1 CN=c1[nH]c(C(=O)OCCOCc2cccc(Cl)c2)cs1 C1(NC(C(CN(C)C)O)=O)C2CCC(C2)C1C(=O)NC1CC2CC1CC2CO N=c1nc(C(=O)NC2(C(=O)NCCOc3ccccn3)CC(O)C2)[nH][nH]1 C(=O)(CC(C(C)C)NC(C1(F)CCC1)=O)NC(c1scc(C)n1)C c1(N2CCN(c3c(C)nsc3)CC2)ncnc(N2CCCC(CNC)C2)c1C c1(C(N2CC(CNC(C(C(C)(C)C)O)=O)C2)=O)cc2c(cn1)OCCC2 C1(CNC(=O)Cn2ncnn2)CC2(CCOCC2)CN1C(c1cc(Cl)on1)=O C1(F)(C(=O)NC(C(=O)NCC2CN(C(C3(c4ccsc4)CC3)=O)C2)=O)CCCC1 c1(C(N2CC3(C(NC(C(CCC)C)=O)CC3)C2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 Cc1cc(-c2cn(Cc3ccc(C(=O)NC4(C)CC4C)o3)nn2)ccc1F C1(CNC(C2CC=C(C)CC2)=O)CN(C(c2cccc(N)c2C)=O)C(C)(C)C1 c1(C(N2CC3C(Cc4cc(C)c(Cl)nc4)C3C2)=O)cccc2cncc(Br)c12 N1(C(CC(=O)OC)=O)CCC2C1CCCN2C(=O)CCc1ccc(N(C)C)cc1 CC(F)(F)C(C)(C)CC(=O)NC1CC(CNC(=O)Cc2n[nH]cc2Br)C1 N1(C(C(c2ccc(C)cc2)C)=O)CC(CNC(=O)Cc2cn[nH]c2)CC(C)(C)C1 c1(C(=O)NC2C(CNC(c3ccc(OC)cc3Cl)=O)C2)ccc2c(c1)OCCO2 CN=c1[nH]nc(CC(=O)N(C(C)CCNC(=O)C(C)(C)c2ccn(C)n2)C)s1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC(CCCCNC(c2ccoc2C)=O)C1 C12CC3(CCC(CC3)C(=O)N1)C2.Cc1n[nH]c(=NCc2cccc(CO)c2)o1 CCCC(CCC)C(=O)NC(C)(CSC)C(=O)NC(C(C)C)C1CC1 C1(C(=O)NC2CC3(CCC3)C2)(NC(c2cocn2)=O)CCOCC1 C1(NC(N(CC(C)OC)C)=O)CNc2c(c(C)nn2C)C1 c1(C(N2CC(NC(c3nnn(C(C)(C)C)n3)=O)C(F)C2)=O)cncc([N+](=O)[O-])c1 c1(C(N2CC(C)(NC(C(C)SC(C)C)=O)C2)=O)ccc2cccc(F)c2n1 N1(C(C(CC)OCC)=O)CCC(C)(CC(N2CCC(CC3CC3)C2)=O)C1 C1(NC(C2CC(F)(F)CS2)=O)C2CC1N(C(=O)CCc1ccncn1)C2 N1(C(C2(F)CN(C(c3c(OC)noc3C)=O)C2)=O)CC2CC1CN2C(C)C c1(C(=O)NC(c2ccccc2)CNC(C2(OC)CC2)=O)cc2cc(F)ccc2o1 C(C(CC(F)(F)F)NC(C1C2(CC2)C12CC2)=O)NC(c1c(C)nc(O)s1)=O N1(C(C=CC=CCC)=O)CCC(C)C1C(=O)NC(C)C(C)SC CC1(NC(=O)C(Cc2ccoc2)NC(C2C=CCS2)=O)CCCOC1 C(=O)(CCCNC(=O)C(C)CNC(C1C=CCS1)=O)OC C1(n2c(-c3nccc(SC)c3)nc(-c3ncccn3)n2)CC(C)(C)OC1=O C=CCCC(C)N=c1nc(N2CCCC(N3CCCC3)C2)c2c([nH]1)CCCCC2 c1(C(N2C(C)(C)C(CNC(c3ccco3)=O)CC2)=O)snc2ccc(Br)cc12 C(=O)(C(C(C)(C)C)C1CCC1)NC(C)CCN(C)C(c1cnn(CC2CC2)c1)=O C(C)(CCCNC(=O)C(C)(C)c1nncn1C)NC(COC(CC)C)=O N1(C(CC(C=C)C)=O)CC2CCN(C(c3c4c(nn3C)CCSC4)=O)CC(C2)C1 C1(NC(CC2(C=C)CC2)=O)CCN(C(c2c(C)ccc3n[nH]cc23)=O)CC(C)(C)C1 C=CCC(CNC(=O)CN(C)C(C1CCC(C)(O)CC1)=O)CC(C)C c1(C(=O)NC)cccc(C(N2CCCC2C(C)NC(=O)CCC2(C)CC2)=O)n1 C1(C(C)C)CN(C)CCN1C(=O)N(CCOc1ccc(Cl)nc1)C1CC1 C(c1ccccc1)=CC(N1CC(C)C1C(=O)NCC(C)(C)C1CC1)=O c1(NC(C2CC(NC(c3nc4ccccn4n3)=O)C2)=O)nccc2cccnc12 CCC(C)(C)CC(=O)N(C(C)CNC(=O)CC1CC(N(C)C)C1)C c1(NC(N2C(CN=[N+]=[N-])CCC2)=O)ccc(C23CCC(C2)NC3)cc1 C12(NOC(=O)CC3CCCCC3F)CCC(NC(=O)CCc3cnn[nH]3)(CC1)C2 Cc1ccc2c(CC(C)Nc3noc(C4CC4)n3)c[nH]c2c1 n1(CC)nc(Br)cc1C(C(=O)NC1(C)CC1)N(C)CC1CC2(CC2)CO1 [N-]=[N+]=Nc1ccc(NC(=O)CC(CC2CC2)NC(=O)CC2CCC2)cc1 Cc1c(C(=O)NCC(C)(C)CNC(=O)C(C)n2cccc2)cccc1F c1(C(=O)NCC(CCNC(C2(Cl)CC2(F)F)=O)OC)cncc(C)n1 C(=O)(CCCCC1CC1)N(C1CC(NC(C2CCN2C2CCCCC2)=O)C1)C c1(C(N2CCCC(NC(=O)NC)C2)C(=O)NC2COC2)c[nH]c2ccnc(Cl)c12 C1(n2c(-c3ccc(C)nc3C)nc(-c3scc(C)n3)n2)CCC2(CC1)CC2(F)F N1(C(c2c(CCC)occ2)=O)CC2(COC(CNC(=O)C(O)C(C)C)C2)C1 c1(C(=O)NC(CC=C)CNC(C2CNC(=O)N2C)=O)[nH]nc2ncnc(O)c12 C1(C(N2CC(C)(OCC(=O)NCCc3ncon3)C2)=O)CCCNC1=O CC(C)C(O)C(F)(F)C(=O)NCCN(C(=O)C1=CCCC1C)C1CCCCCC1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(CCCNC(CC(CC)C)=O)C N1(C(C(C)NC(N)=O)=O)CC2CC(NC(=O)CCCc3cnn[nH]3)C1C2 C1(CC(N2C(CN(C(=O)CCCF)C)CCC2)=O)CCc2sccc2C1=O c1(OC)ccc2c(c1)C(C(=O)NCCC1(NC(C3(O)CCSC3)=O)CC1)CO2 CC1(CNC(c2cocn2)=O)CCCN(C(C23CC(CO)CC2C3)=O)C1 C1(CNC(C2C(=O)NCC2)=O)CCCCN(C(C2(O)CCCCC2)=O)C1 N1(C(CC2CCC(=O)NC2=O)=O)CC2COCCC2(NC(=O)C=CC2CCC2)C1 c1(CNc2cc(Br)ccc2C(CO)OC)cc(Br)cc([N+](=O)[O-])c1O C1(C#CC(=O)NC2(C)CN(C(=O)Cc3ccc(Br)s3)C2)(CC)COC1 N1(C(CCc2cn(C)nn2)=O)CCC(CNC(=O)CC2CC3C=CC2C3)CC1 CCCCC(C)(F)C(=O)N1CC(CCNC(c2ccc(N=[N+]=[N-])cc2)=O)C1 N1(C(CC)=O)CCN(C(=O)C(O)CC2CCCCC2)C(C2CCC2)C1 C12(CN)CCC(C(=O)NCC(c3n[nH]cc3[N+](=O)[O-])(F)F)(CC1)C2 c1(C(=O)NC2CCN(C(=O)CC3C=CCCC3)C2)cnc(S)nc1 c1(CNC(C(=O)NCC)=O)cnn2c1C(=O)NCC2.c12ncccc1CNC2=O C1(CNC(=O)COCC(c2ccccc2)=O)CN(C(c2nncs2)=O)CC12CC2 C1(C(C)C)CN(C(=O)C(C)(C)N2CCCC2)CC1C(=O)NC1CC(F)C1 N1(Cc2c(CCCC)cccc2)CCC2(NC(=O)Cc3sccc3C)CCCC12 CCCCCC(C)CC(=O)NC1CC2CCC(C1)N2C(C12CC1COC2(C)C)=O c1(COC)nc(NC(COC)C2(C)CC2)cc(=NCc2cccc(N)c2C)[nH]1 C1(O)(CNC(C(CC)OCC)=O)CCN(C(c2n[nH]c(C)c2F)=O)C1 C1(CNC(=O)Cc2cc[nH]c2)CC2(CC2)CN1C(C1CCSCC1)=O C1(CNC(c2cccs2)=O)CC12CCN(C(=O)CSc1c(C(C)C)con1)CC2 C(C(C)CC(=O)N1CCOC(CN(C)C(c2cc(C(C)(C)C)no2)=O)C1)OC C1(OC)CC(C(=O)Nc2ccc(Cl)cc2)N(C(=O)CCc2cncs2)C1 C1Cc2[nH]c(=NCC34CCC(CC3)C4)[nH]c(=NC3CC(=C4CC4)C3)c2CO1 C1(C)(CNC(c2cc(C(C)C)on2)=O)CCCN(C(=O)CC(F)(F)Cl)C1 c1(C(N(C)CC2C3CN(C(C(C4CC4)SC)=O)CC32)=O)ccc(SC)cc1C C1(C(N2C(C)CC(NC(C3C4CC5C(C4)C35)=O)CC2)=O)CC2CC1CC2(F)F C1(CNC(c2ccn(C)n2)=O)CCN(C(C2C(C#N)C2(C)C)=O)C12CCC2 C1(CCNC(=O)C=CCO)CN(C(c2ccc(F)s2)=O)CCO1 C=C=CC(C)C(=O)NCC(N1CCN(C(c2cc(Br)n[nH]2)=O)CC1)C C(C(=O)NNC(=O)C(C)c1ccccc1)c1cc(-c2cccc(OC)c2)on1 C(=O)(C(C)CC(C)(C)C)N1C(CNC(CCC(C)OCC)=O)CCC1 c1(C(N2CCC(CC(=O)NC(c3ccccc3)C(C)C)C2)=O)ncn2c1CCC2 N1(C(C(C)SC(C)C)=O)CC(CC(N2CCNC(=O)C2CCO)=O)CC1(C)C CCCCC(C)C(=O)N1CCOC(C)C1C(=O)Nc1cncnc1C C1(NC(COC(CC)C)=O)(CO)CCN(C(c2ccc(C(C)=O)s2)=O)C1 C12(C(N3CC(NC(C4(C)CC(=C)C4)=O)C3)=O)CC(CO)(C1)OC2(C)C C(=O)(N=c1[nH][nH]c2cccnc12)C1(C)N(CC)CC1.c12nn(C)cc1NC2=O N1(C(C2CC3C(C)(C)C3C2)=O)CC2(CCC(NC(C34COCC(C3)C4)=O)CC2)C1 CN1CCCC(F)(C(=O)NCC2CCN(C(C3(C)CCOCC3)=O)C2)C1 c1([SH](CC(=O)N(C(=O)C2=C(C)CCCC2)CCC)NCC)ccc2c(c1)CCC2 c1(SCC)ccc(-c2cn(CC3CCCCN3C(=O)C(C)C(F)F)nn2)cc1 Cn1cc(N)c(C(N2CC(F)(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)n1 C1(NC(c2n(C)c3c(n2)cccc3)=O)COC2(CCN(C(C3CCC3)=O)C2)C1 C1(O)(CCNC(c2ccc(OC)nn2)=O)CCCN(C(c2cncc(O)c2)=O)C1 N1(C(Cc2cc(C)on2)=O)CC2(C(=O)NCCc3cn[nH]c3)CC1CCO2 C1(CNC(C=CC(CC)=CC)=O)(CNC(C2C3CCCCC23)=O)CCCCC1 C=CC(COC)N=c1nc(N2CCc3oc(C)nc3C2)c2ncccc2[nH]1 Cc1cccc(C)c1C(N1CC2CC2(CNC(c2ccncc2)=O)C1)=O C1(O)(CNC(CC=CCC)=O)CCN(C(=O)CNC(c2ccccc2F)=O)CC1 C(C(=O)N=c1ccn(CC2CC2)[nH]1)C1N(C(CCCC(=C)C)=O)CC(O)C1 N1(C(C(C(C)C)CO)=O)C2CCCC1CN(C(=O)C=CCCC(F)(F)F)C2 C#CC(C)(C)C(=O)NC1C=CCN(C(C2CC(=O)C2(C)C)=O)C1 N1(C(C=CC(=O)OCC)=O)CCSCC1CCNC(=O)CC1CCC2CC2C1 CCC(C(=O)NCC(C)(C)OCC(=O)NCC1CCOC(C)(C)C1)C(C)(C)CC N1(C(CNC(c2c(C)cns2)=O)=O)CC2CC(NC(c3ncccc3Cl)=O)C1C2 c1(C(N2CC(OC)C(NC(=O)Cn3cnnc3O)C2)=O)nn(C)cc1S(N)(=O)=O c1(NCC2N(C(C(c3c(C)cccc3)(C)C)=O)CC2)snc(Cl)c1C#N N1(C(C=CC(C)=O)=O)CCCC(CNC(=O)Cc2cnc(C)[nH]2)CC1 C1(CNC(C(C)(CC)OC)=O)C(C)CCCN1C(=O)CC=Cc1ccc(F)cc1 N1(C(c2nc(C)c(C)s2)=O)CCC(CCNC(C23CCCC2C3)=O)C(F)(F)C1 N1(C(C=C(CC)C)=O)CC(OC)C(NC(c2cncc(COC)c2)=O)C1 c1(C(=O)NC2COCCN(Cc3cccc(Cl)c3)C2)ccc2nnc(S)n2c1 c1(CNC(N2CC3(C(C(=O)OC)C3)C2)=O)cc([N+](=O)[O-])c(O)cc1N C1(CNC(C(C)NC=O)=O)(NC(C2CCCC(CC#N)C2)=O)CCCCC1 CCCC(C)(C)C(=O)N1CC(CNC(=O)CCSCC)C1 Cc1cn2cc(NC(C3CC4(CC4)CN3Cc3ccc(Br)cc3C)=O)ccc2n1 C1(CNC(C(CC)OC)=O)CN(C(=O)CCNc2c(C)noc2C)CC1O c1(C(N2CC(NC(CCC3CCC(OC)C3)=O)C(C)C2)=O)cc([N+](=O)[O-])oc1C C12(NC(c3nc(COC)sc3)=O)CCCC1N(C(=O)CCc1ccnn1C)CC2 c1(C(=O)NCCC(C)N(C(c2c(OC)ccc(O)c2)=O)C)cnc2sc(C)cn12 O=C(O)C(CC(F)F)NC1CC2CCCC1C2 C1(c2cc3[nH]c(=N)oc3cc2)NC(=S)N(c2ccccc2)C2=C1C(=O)NC21CCOC1 Cn1c(=O)cc(-c2noc(CCc3cccc(F)c3)n2)c2ccccc12 N1(C(C(C)C(C)C2CCCCC2)=O)CC(NC(=O)C(F)=C2CCC2)C(C2CC2)C1 c1(C(=O)NCCC(CCn2cc(CCCSC)nn2)(F)F)ccnc(Br)c1F C1(C(=O)NCCC2(OC)CN(C(c3conc3C)=O)C2)CCc2nc(C)cn2C1 c1(OC)ccc(OC)c(CC(C)NCc2ccnn2C2CCCCO2)c1 c1(OC)ccc(C(N2CC(CC)N(C(C3CCCC3)=O)CC2)=O)c2ccncc12 C=CC(CC)CC(=O)N1CC2CC2(NC(=O)C(c2cccc(Cl)c2)(C)C)C1 C1(C(=O)NCCC(C)C)C2CCCC1CN(Cc1cccc(Cl)c1F)C2 C1(C(C)O)CCC(NC(C2(N(C)C(c3c[nH]c(=N)o3)=O)CC2)=O)CC1 c1(C(=O)NCCC2CN(C(C(CCC)C)=O)CC2C)nccc(C)c1N CC(C)CC(C)(C)C(=O)NCC12CC(NC(C3CCSCC3)=O)(C1)C2 c1(NC(C2N(Cc3nc(C)c(Br)cc3)CCN(C)C2)=O)ccc2c(c1)CCC2 CCC(CNC(=O)C(C)Oc1cccc(F)c1)(CC)NC(=O)CCCN(C)C N1(C(COCCS(C)(=O)=O)=O)CCN(C(c2ccc(C(=O)CF)cc2)=O)CC1 c1(C(N2CCCC(NC(C3CN(CCOC)C(=O)C3)=O)C2)=O)cc(C)c(C)nn1 c1(C(=O)NC2C(CNC(CN3CC(OC)C3)=O)OCC2)ccn(C)c(=O)c1 C(=O)(C#CC1(C)CCCO1)N1CCN(C(CCC(C)(C)F)=O)CC1CO c1(C(C)OC(c2ccc(CC#N)cn2)=O)ccc(-c2ccccc2)nc1 Cc1cc(NC(=O)C(C)NC(=O)C(N2CCNC2=O)C)cc(C)c1F CCC(C(=O)NC(C)CCNC(=O)CCCSC(C)(C)C)SC c1(OC)ccc(CC(=O)NC(CNC(c2c(C)nnn2C)=O)C2CC2)nc1 Cc1c(C(=O)N(C)CC2CCCCN2C(=O)C(C)C2CC2)cccc1S(N)(=O)=O c1(CC(=O)NCC(C)NC(c2ncn(C)n2)=O)ccnc(F)c1F c1(OCC)cccc(-c2cnc(CNC(=O)NCC3(C)CCC(=O)N3)cn2)c1 CCCC(CCCNC(=O)C(=Cc1ccncc1)C)NC(=O)C(C(C)C)C1CC1 N1(C(C)=O)CCC(C)(C(=O)NCC(C2CC2)N(C(=O)CSc2nc[nH]n2)C)C1 C1(N(C2COC2)C(C)=O)CCCCC(=O)N1.C1(=O)C(CC2CCCC2)N1c1cncnc1 c1(C(N(CC(C)(C)CNC(C2(O)COC2)=O)CC)=O)ccc(C)c2ncccc12 C(C(C)(O)C(C)(C)C)NC(=O)CCCC1CCCO1.CC12CN(C1)C(=O)CC2 C1(O)(CNC(CN(CC(C)(C)C)C)=O)CCN(C(=O)C(C2CCOCC2)C)CC1 C1(CNC(C2C(C(=O)OC)C2)=O)CCCC2CN(C(=O)C(C)C3CC3)CC12 c1(C(N(C)CC2(NC(=O)CCc3ccco3)CC2)=O)cc2n(c1)CCOC2 CCCCC(=O)NC(COC(C1(CSC)CC1)C)CO C1(C(C)(O)CNC(=O)Cc2cnc(C3CC3)[nH]2)CCN(C(c2cnco2)=O)CC1 C1(O)(COC)CCN(C(=O)CN(C(=O)CC2C=CCC2)CO)C1.C1(CN)CC1 C(=O)(CN=Cc1ccco1)N1CCC(O)(C(=O)NCc2ncn(C)c2)CC1 N(C(=NCCCn1cccn1)NCC(C)C)C(CC)C(F)F c1(C(N2CCN(C(c3cncc(OCC)c3)=O)CC2C)=O)cc(Cl)cc(F)c1Cl C1(N(C(c2csc(N3CCCCC3)n2)=O)CC)CCN(C(c2ccsn2)=O)CC1 CCCN=C(NCCOC(C)(C)C)NC(C)CNC(C1CCCCC1)=O CCCCS(=O)(=O)CC(=O)N1CC2CC1CN(C(=O)Cc1cccs1)C2 N1(C(CC(=O)NCC)=O)CCCC(C(=O)Nc2cc(C(=O)OC)cc(Cl)n2)CC1 c1(C(N2CCC(n3cccn3)C2)=O)cc(=O)c2ccc(C3CC3)cc2o1 c1(C(N2CCCC(C(C)NC(CCCC#CC)=O)C2)=O)ncc(C#N)cc1C O=S(=O)(c1c(Cl)cccc1Cl)N1CCn2cccc2C1.C1(N)CC12CCNCC2 N1(C(C2CCCN2C(c2ccsc2)=O)=O)CCCc2cc(F)c(F)cc21 N1(C(C=CC(CC)=CC)=O)CC2CCN(C(=O)C(F)(F)COC)CCC2C1 CCCCC(=O)C(=O)N1CCCC(CCC(=O)N(C2CCCC2)CCO)C1 c12nc(cs1)C(=O)N2.C1(CC(=O)OC)CCN(C(=O)COC2CCN(C)C2)C1 Cc1nccnc1C(C(=O)NCC(C)(C)CC1CCCO1)N(CCSC(F)F)CC C(=O)(C1=NOC(C)C1)N1C2C(CNC(CCc3c(C)nccc3)=O)C(C2)C1 C1(C)(C(=O)NCC(CCC)NC(=O)C(C)(C)COC)CCCCC1 CC(C)(C)C(O)Cc1cn(C2CC2)nn1.N12CCCC(C1)CCNC(=O)CC2 C1(CCC(=O)N(C2CC(F)(F)C2)C)(C(=O)NCC2CC2Cl)CCCC1 C1(C(N(CC(CC)OC)C)=O)CCCN(C(=O)CN2CC(C)(OC)C2)C1 c1(CC(N2CC(CNC(C=C(CCC)C)=O)OCC2)=O)c(CC)nn(C)c1CC C1(NC(c2cccc(=O)o2)=O)COC2(CCN(C(c3ccncc3Cl)=O)CC2)C1 C=CC1OCCC1C(=O)C(C(C)C)c1cnc(C)s1 C1(N(C)C)CCCC1NC(=O)CN.C12CC(C1)C(=O)NC2.C1(C(=O)NC2CC2)CCC1 C12(NC(CCCC(C)=O)=O)CN(C(C3CC=CC3)=O)CC1CS(=O)(=O)C2 N1(C(C=CCN(C(C(C)CCN(C)C)=O)C)=O)CCC(O)C12CCC2 c1(C(N2CC3(CCC(CNC(CCC(=C)C)=O)O3)C2)=O)cc2cc(F)ccc2s1 Clc1cc(-c2cc(Cn3cccn3)on2)cs1 N1(C(CC)CNC(c2cnn(CC(=O)OC)c2Br)=O)CCOC(C2CC2)C1 N1(C(=O)NC(C)C(=O)Nc2ccccc2SC(C)C)CCC(C)(C(=O)N)C1.CO N1(c2nnc(C(C)C)n2CCCN2CCCS2(=O)=O)CC(=O)N2CCCCC2C1 c1(C(=O)NC(CC(C)NC(C2(CO)CC(C)(C)C2)=O)C)[nH]ncc1C#N C1(NC(C2CCC=CO2)=O)CN(C(=O)Cc2cccc(C(F)(F)F)c2)CCC1O N1(C(C(C)(C2CC2)OC)=O)CC2CN(C(=O)Cc3cccc(C)c3Cl)CC2C1 C#CC12CC(CN1C(C1COCCN(C(=O)C3=C(C)CC3)C1)=O)C2 N1(C(Cc2n[nH]c(=NC)s2)=O)CC2(C1)CN(C(C1CCS1(=O)=O)=O)CCO2 C1(OC)CN(C(=O)CCn2cccn2)CC1NC(c1ccsc1C(F)(F)F)=O C1(NC(c2cc(OC)c(O)nc2)=O)CCCC2CN(C(=O)Cc3ccsn3)CC12 C1(CNC(=O)CCc2ccnc(Cl)c2)CC2CCC1N2C(c1ccsn1)=O N1(CC)CCOCC1C(=O)NCCCN(C(c1cc(C)c(Br)s1)=O)CC c1(CCC(=O)NCCCCC(C)NC(C(C)OCOC)=O)ccc(Cl)c(F)c1 CP(C)(=O)CC(=O)NCCC1(O)CN(C(C2(C3CC3)CCCO2)=O)C1 c1(C(=O)NCCCCn2cc(C(C)(C)NC(C)C)nn2)ncn2ccccc12 CC1(C)CC(CNC(=O)CCNC(c2ccoc2)=O)N(C(=O)CC2COC(=O)C2)C1 N1(Cc2ccc(OCC(=O)OC)cc2)CC(C)CN(C(=O)C2=CCCC2)CC1C C1(SCC)CCCCC1NC(C1(CNC(=O)CCc2cocn2)CC1)=O CCC(CC(=O)NCC12CC(NC(=O)C=C(C)C(C)C)(CO1)C2)C1CC1 N1(C(CC#N)=O)CC2CCN(C(c3cnc(-c4ncccn4)s3)=O)CC2C1 c1(OC)cc(C(N2CC(C(N3CCC(F)CC3)=O)CC(C)C2)=O)cc(Cl)n1 C(=O)(C1Cc2ccccc21)NC1(C(=O)Nc2c(CC)nc(C)cc2)CSC1 Cn1cc(C(=O)NC(Cn2cncn2)C(N2CC(C)(C)C2C2CC2)=O)ccc1=O N1(C(c2[nH]c(=NCC)sc2)=O)CCc2ccc(C)c(Cl)c2C1 C(=O)(CC1CCC(=O)c2ccccc21)NCC1N(C(C(COC)COC)=O)CC1 c1(C(N2C(CN(C(c3noc(CC)c3C)=O)CC)CCCC2)=O)ccc(O)c(F)c1 c1(CN2CCCC(NC(c3ccnnc3O)=O)C2)cc(F)c(Cl)cc1Cl c1(NC(CC2CN(C(C(CC)O)=O)C2)=O)cnccc1C C(CCCCC(=O)NC(CCNC(c1nccc(SC)n1)=O)C(C)C)OC CC1CC(O)CN(C(=O)C(CCN(C)C)NC(c2nc(=N)cc[nH]2)=O)C1 C1(C(=O)NC(CNC(C(C)OCCOC)=O)CO)CCN(C(=O)NC2CC2)CC1 c1(C(=O)NC2CCC(CNC(C(C)CC3CCC3)=O)C2)nn2cccnc2c1Cl C1(C(N(CCCN(C)C(C2CC3CC2C3)=O)C)=O)CCCCN1S(N)(=O)=O C(CCC)(C(O)C(=O)NCCN1CCC(CO)C1)NC(C1C(=C)C1)=O C#Cc1cc(F)c(C(=O)NCCCN(C)C(c2cncn2C)=O)c(F)c1 C1(NC(c2cnc(C)o2)=O)CCCC(NC(=O)Cc2csc(N(C)CCO)n2)C1 C(C(C)(O)CNC(=O)CSCc1ncc[nH]1)NC(COCCC)=O CCC(CC)(C(=O)NC1CN(C(c2cc(C)nn2C)=O)CC1n1ccnn1)OC n1(CC)ncnc1C(N1CCCC1CCNC(c1cnc(N(C)C)s1)=O)=O CC1CCN(S(=O)(=O)c2cnccc2N2CCC(n3ccnn3)C2)CCC1(F)F c1(CC)cccnc1C(=O)NCC(C1CCN(C(c2nccn2C)=O)CC1)C C(C)(CO)(C(=O)OC)N(C(=O)CN(C)CC1CCCO1)Cc1cccc(Cl)c1.CO Cc1c(C(=O)NCC2CCCN(C(C34CC(C#N)(C3)C4)=O)C2)cncc1F Cc1cc(C(=O)N(C(C)CN(C)C(c2cc(Cl)no2)=O)C)cc2nn[nH]c12 C=CCC(CO)NC(c1nc(Br)cs1)c1nnnn1C1COC1 N1(C(C)C)CCN(C(C(=O)NC2CCOC2)C(C)C2CCC2)CC1 N1(C(=O)OC(C)(C)C)CC(CC2(C(C)(C)NC(C)=O)CC2)C(F)C1 N1(C(CCOC2(C)CN(C(C(C)(C)O)=O)C2)=O)CCCC2CNC(=O)C12 N1(C(C2CCN(C(CC)=O)C2)=O)CCCCC(NC(=O)C(C)(C)CCCF)CC1 C(=O)(CC(C)(C)O)N(C1CCN(C(=O)CNC=O)C1)CCC C(=O)(C1=CC2(CCOC2)C1)N(C)CC1COCCN1c1ccnc(C(C)(C)C)n1 C1(NC(c2c(N)non2)=O)CCCCC1NC(c1csc(N2CCCCC2)n1)=O C1(NC(c2ccc(CC)[nH]2)=O)CCC2CN(C(=O)Cc3cncnc3)CC2C1 C1(C(N(CC(C)N(C(=O)CCOC2CC2)C)C)=O)CCc2c[nH]nc2C1 N1(C(c2c(C)[nH]cc2)=O)CCC2CN(C(=O)CNS(=O)(=O)c3cccs3)CC12 CC(C)C1=NOC(C(=O)N(CCCNC(=O)C(C)N2CC(C)C2)C)C1 c1(C(N2CCN(C(C(C)CC3CC3)=O)CC2C2CCC2)=O)cc(F)cc(N)c1F CC1CCCCCC1NC(=O)CN(C)C(C1CC(C(C)(C)C)=NO1)=O C12(CCSCC1)C(=O)O2.c1(NC(C(C)NCC)=O)ccncc1OC C1(C(N(CCOCCCNC(C2CCC(CC)CC2)=O)C)=O)CCCS(=O)(=O)N1 C1(NC(c2ccc(OCC)c(F)c2)=O)CCc2cc(OC)ccc2C1 C1(NC(CC(c2c(C)cccc2)C)=O)CN(C(=O)C(C)c2ccsc2)CCC1C C1(NC(C(n2c(C)cc(C)n2)C)=O)CCC2CN(C(c3cnsc3C)=O)CC2C1 N1(C(C=Cc2n(CC)ncc2)=O)CCC2(CC1)CC2CNC(=O)Cn1cncn1 C(C1CCc2nccn21)NC(C1CC12CCN(C(c1cccc(O)c1F)=O)C2)=O C(=O)(C(C)(C)C(C)(F)F)N(C)CC1CN(C(c2cn(C)nc2C2CC2)=O)CCO1 c1(NC(N(CCCC)C(C)CC)=O)ccc(-n2c(C)ccc2C)cc1 c1(OC)cc(C(=O)NCC(C)NC(=O)C(C2CCCCCCC2)O)ccc1Cl CC(C)C(C)C(CNC(=O)C(c1ccccc1Cl)O)N=c1ccc(C#N)c[nH]1 N1(C(C2CC(C)(CC)C2)=O)CCC(CNC(c2cc(C)cc(C)n2)=O)C(O)C1 C1(COC)CN(C(c2n[nH]cc2I)=O)CCN1C(C1CCCO1)=O CN(S(=O)(=O)N1CCCCC(C)C1)CC(=O)OCCl.C(C)(C)C C1(CC)CN(C(=O)C=CC(C)(C)NC(=O)C(C)N(C)C)CCO1 C(=O)(C1=CCC2CCC1N2C(=O)CCCc1cnn[nH]1)N(C(CSC)C)C C1(C(N2CCC(C)(NC(c3ccc(C(=O)OC)[nH]3)=O)C2)=O)CCC(N=[N+]=[N-])C1 CN1CCCCC(C(N2CC(CNC(=O)C(F)C(F)(F)F)C2)=O)C1=O CN1CCCC(CNC(C2CN(C(C3CC(F)(F)C3)=O)CC2(F)F)=O)C1=O CC12COC(C(N3CCCC(NC(C4CC(CC5CC5)C4)=O)C3)=O)(C1)C2 CC1C(C(F)(F)F)CCN1C(C1CCCCCC1)C(=O)NC1CCOC1 c1(C(=O)NC2CCCC2CNC(C2CC2C(F)(F)F)=O)cncc(C2CC2)c1 Cc1cc(C(N2CCCC(C(=O)Nc3cccnc3C#N)CC2)=O)cc(C#N)c1 CCC(CC)C(C(=O)NCC1CCC(F)(CNC(=O)C(C)(C)F)C1)OC CN=c1cc(C(=O)NC2CCN(C(c3cccn3C3CC3)=O)CC2CO)cc[nH]1 Cc1nn(C)cc1C(=O)N(C(CNC(c1nc(Br)c(C)s1)=O)C1CC1)C c1(C(N2CCC(O)(C(C)NC(=O)Cc3nncs3)CC2)=O)ccc2scnc2c1 CC(C)CCC(=O)NCc1cnn(C)c1C(=O)NCC(Cl)Cl c1(CN(C(C2(C3CC3)CCCO2)C(=O)NCCCC)C)ccc2cc[nH]c2c1 C1(CC)CC2CCC(C1)N2C(C1(F)CCN(C(c2cncn(C)c2=O)=O)C1)=O c1(C(=O)NCC(CC=C)NC(C2CNC(=O)N2C)=O)cnn2c(N)cc(C)nc12 N1(c2n(C3CCC(C)C3)c(-c3ccc(Cl)nc3)nn2)CC2CCC(=O)NC2C1 CCCC(CCCO)C(=O)NCC1CC(C)(C)CN1C(=O)CC1CCC2CC12 CCCCC(CC)CCC(=O)N1CCC(NC(=O)C(C)NC(=O)C2CC2)C1C N1(C(C(C)N2CCC2)=O)CC2CCC1C2NC(c1cc(C2CC2)n(C)n1)=O C(=O)(C(CC)(CC)CC(=O)OCC)NC1CN(C(C2CC(C#C)(O)C2)=O)CC1C C(CC(C(=O)N(CC(C)(CO)CO)C)NC(=O)CN(C)C(=O)NC1CC1)=CC N1(C(CC)=O)CCCC1C(=O)NC1CC1(C)C c1(N2CCN(C(C(=O)Nc3cccc(Cl)c3Br)=O)CC2)nc2ccccc2s1 C#Cc1cc(C(=O)NC2CN(C(c3cccc(C(F)(F)F)c3C)=O)C2)cc(F)c1 c1(C(=O)NC2CC(NC(CN(C(=O)OC)C)=O)C2)[nH]c2ccc(F)cc2c1C C1(NC(C2C(COC)C2)=O)CCCN(c2cc(C)nn2C)C1=O C=CCC(CNC(C1COCCN1C(=O)C(C)CO)=O)CC(C)C N1(C(CC2(CSC)CC2)=O)CCC(C(=O)N(C)Cc2ccc(O)cc2)CC1(C)C C1(C)(CCNC(C(CC)n2cncn2)=O)CCN(C(=O)CS(=O)(=O)NC)C1 CC(C)C(C(=O)NC12CCC(CNC(C3CC3c3ccco3)=O)(C1)OC2)C(C)C c1(C(c2n(CCOCC)nnn2)Nc2ccc(C3CC3)cc2)c(Cl)cccc1Cl c1(CN2CCC(N(c3ncncc3C#N)C)C2)cc(Cl)ccc1Br CC(C)CC(CNC(=O)CCN(C(=O)CCCC(=O)C1CCC1)C)CO CC1C2CC(C2NC(=O)C(c2cccnc2)O)N1C(C1CC(C)(C)C1)=O c1(-c2cn(C)nc2)cncc(C(=O)NCC2(O)CCN(C(=O)CNC=O)C2)c1 N1(C(c2cccc(C(C3CCC3)OC)c2)C(=O)NC2(C)CC2)CC2OCOC2C1 c1(C(N(CCC(C)NC(c2ccc(Cl)s2)=O)C)=O)ccc(C(F)F)nc1 n1(C(CC)C)ccc(=NC(=O)C23CCCC2CCN3C(=O)CNC(N)=O)[nH]1 c1(C(N2CCC(C(C)NC(=O)CN(C)CC3CCCC3)C2)=O)ccccc1Cl C=CC(CCC)CC(=O)NCC(CO)NC(=O)CCOc1ccccc1Br CC1=C(C(=O)N2CCCC(C)(NC(=O)Cn3cc([N+](=O)[O-])cn3)C2)CCC1 C1(CNC(=O)Cc2sc(O)nc2O)CC(NC(c2cccc(=O)o2)=O)C12CCC2 C(=O)(CC(C)(C)C(F)(F)F)N(CC(CNC(COCCCCC)=O)O)C1CC1 n1(CCCOCC)c(N2CCC(C)C2C(=O)O)nnc1-c1ccc(Br)s1 Cc1nccc(Br)c1NC(C1CC1NC(=O)Cc1cccc(Cl)c1F)=O C(CCCCCN=C(NCCCC1(C)CC1)NCC(C)(C)C1CCCO1)SC CCS(=O)CC(=O)NCc1cn(C2CN(C(C)C)C2)nn1.C1(C=O)C2CC3C(C2)C13 CC(C)C(O)C(F)(F)C(=O)NC(C)CCCCNC(=O)CCc1cccc(O)c1 CC(CC(=O)NCC1(OC(C)C)CCC1)C(C)(C)NC(c1ccncn1)=O C(CC(O)CNC(C1CCOC1=O)=O)NC(C1(CC#C)CCC1)=O C1(C(=O)Nc2c(N(C)C)nccc2)CCC2CCC1N2C(c1cc(CO)on1)=O O=[N+]([O-])c1cccc2c(N(C3CC4CNC3C4)C(C34CC(C3)C4)=O)ncnc12 C(CC(=O)N1CCC(C(=O)NCc2nonc2C)O1)c1c(OC)cnn1C C1(=O)C(Cc2ccoc2)O1.C1(C(NOC(C=C)C)=O)OCCC1C(=O)OC N1(C(C2(CSC)CC2)=O)CC2CCOC2(CNC(=O)C(CC)N(C)C)C1 N1(C(C2=C(SC)CCCC2)=O)CC2(C)CN(C(=O)C(C)CC(N)=O)CC2(C)C1 N1(C(CS(CC)=O)=O)CCC2CN(C(c3cc(N)ccc3C)=O)CC2CC1 CC1CC2CN(C(=O)CCC#N)CC2N1C(c1ccc(CF)cc1)=O CC(C)(CCCNC(=O)Cc1cccnc1N)NC(C1CC(O)C1)=O N1(C(C2N(C)C(=O)NC2)=O)CCCC(C2CCCN(Cc3ccccc3)C2)C1 N1(C(c2c(C)cccn2)=O)CC(NC(C2CCC(F)C2)=O)C(C2CC2)C1 CCC(CN(C)C)CC(=O)N(CCCCN(C)C(C1CC2(CCCC2)C1)=O)C N1(C(C(CN(C)C)O)=O)CCCCC1C1CN(C(=O)C(=O)N(CC(F)F)CCO)C1 C(=O)(C(C)(F)C(C)(C)F)NC(C(C)NC(C(CC)CC)=O)CO C1(C(F)(F)F)(C(=O)NCC2(NC(CC=C)=O)CCOC2)CC2C=CC1CC2 n1(CC(=O)NCC2(OC)CN(C(C34CC(F)C3C4)=O)C2)nc(C)ccc1=O c1(CNC2C(C(=O)Nc3cnn(C)n3)CCC2)ccc2ccccc2n1 Cc1cncc(C=CC(N2CCCN(C(C3(N4CCCC4)CCC3)=O)CC2)=O)c1 C(=O)(CCN=c1[nH]ccs1)N1C2CC(N(C(C(C)c3ncco3)=O)C)CC1CC2 c1(OCC(C(=O)NCCNC(=O)CC2CC=CCC2)O)ccccc1Cl Cc1cc(C(=O)NCC2CCCC2C(=O)NC2(C(=O)NC3CC3)CC2)nc(O)n1 CSC1=C(C(=O)Nc2ccc(C)cc2)CCCC1.C(=O)(C1=CC(C)(C)C1)NCCCN c1(OC)cccc(OCCC(=O)NC2CC(NC(C3(C)CC3(F)Cl)=O)C2)c1 c1(C(=O)NCC(C)NC(C2CC3CCC2O3)=O)cc2sccc2cn1 c1(OC)ccc(Cl)c(C(=O)NC2(C)CCN(C(C3(SC)CC3)=O)C2)n1 C1(N(C)C(c2cc(C3CC3)cs2)=O)CCCCN(C(=O)CCCCC2CC2)C1 C1(C(=O)NCC(CC(=O)NCC2CC(O)CCO2)OC)(CC)CC(C)(C)C1 Cc1[nH]c(C#N)cc1C(N1CCC(C)C1CNC(=O)C(=O)NCC1CC1)=O N1(c2nnnn2CC)CCCN(C)CC1C.C(C(C)(C)C1CCOC1)NCCC C(=O)(C(C)(C)CS(N)(=O)=O)NCC1C(NC(CCC(=O)NC)=O)C1 Cc1ccc(C(=O)Nc2ccc(CNC(=O)CCc3cccnc3C)nc2)nn1 CCC1=C(C(=O)N(CC(C)CNC(c2sc3cccnc3c2Cl)=O)C)CCCO1 C(CCCCC(=O)N1CCCCCC1C(=O)NCCCCN(C)C)=CC C1(Oc2ccccc2COC)(CN(C)C)COCC1(C)C Cc1ncsc1CC(N1CCCC1CNC(=O)C(n1nccc1C)C)=O C12(C(N3C(CNC(c4ccc(Br)cc4)=O)CCCC3)=O)CCCN1CC(O)C2 C1(CNC(c2cc(CC)c(C)s2)=O)CC2CN(C(=O)C(C(=O)OC)OC)CC12 N1(C(CC(c2ccc(C)cc2)C)=O)CCN(C(C2CC(O)C2)=O)CC1C(C)(C)C C1(C(CNC(C(CC)NC(N)=O)=O)(C)O)CCN(C(=O)CSCC(F)F)CC1 N1(C(C(=O)N(CC(C)O)CC=CCN(C)C)=O)CC2CC3CC2C1C3 N1(C(C2N(C)CC2)=O)CCCC2CN(C(C3CC3C(N)=O)=O)CC12 C=C(C)CC(C(=O)Nc1cccc(CCF)c1)NC(c1cccs1)=O C(CC(=O)NCCc1ccncc1)(C(F)F)NC(c1c(CC)cc[nH]1)=O N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2c[nH]c(=O)cn2)=O)C(CF)C1 Cc1c(CC(=O)NC(C)CC2CN(C(=O)Cc3c(Cl)cnn3C)C2)cnn1C C=C(C)CC(C(=O)NCCC(O)C(=O)N1CC(n2ccnc2)C1)OC C1(CC)CCCCC(c2nc(-c3ncccc3F)no2)N1 c1(CC)sc(=N)[nH]c1C(=O)NC1CC(N(C)C(c2cccnc2C)=O)C1 Cc1cccnc1CC(=O)NCC1CN(C(c2cc(C(F)F)ccn2)=O)C1 N(C1c2ccccc2CCC1C)C(=O)Nc1cc2c(cc1)C(NCC)CC2 C(C(C(=O)NCCCC(C)NC(=O)C(C)SC1CC1)NC(=O)OC(C)(C)C)OC c1(CN2CCC(N(C(=O)CCC3(C)CC3)C)C2)ccc(F)cc1F Cc1cc(C(=O)NC2CCCC23CN(C(C2C=CCCC2)=O)C3)cc(N)c1Cl C(=O)(CN=S(C)(C)=O)NC1CCCN1C1CCCC1NC(c1csc(C)c1C)=O C1(C(C)NC(Cc2c(C)occ2)=O)CCCN(C(c2ncccc2F)=O)C1 N12CC(CC(C)C1)NC2=O.c1(OC(C)C)cccc(SC(F)(F)F)n1 C(CCc1ccc(F)cc1)(C(C)(C)C)NC(C(=O)NC(CC)CSC)=O C1(C(N2CC3C(NC(=O)CCF)C3C2)=O)Cc2cc(F)ccc2O1 C(C(CNC(c1cc2n(c1)CCC2)=O)C(F)(F)F)NC(c1cccc(OC)n1)=O N1(C(COCC(C)(C)C)=O)CCC(NC(c2ccc(Cl)c(F)c2)=O)C(CO)C1 c1(CNC(C(C)Oc2ccccn2)=O)ccc(S(=O)(=O)Oc2ccccc2)cc1F C(=O)(C(C)(C)CC#N)NC(CC)CNC(C1CC1OC(C)(C)C)=O CC1CCN(C(=O)CCc2ccncc2)C(C(N2CCCC(C#N)C2)=O)C1 c1(NCC(=O)NC(C(=O)NCC(F)(F)CO)C2CCCO2)ncccn1 N1(C(C(C)CS(C)=O)=O)CC2(CCN(C(C3CC3Cc3ccccc3)=O)CC2)C1 C1(N(C(C(CCCC)O)=O)C)CC2CCC(C1)N2C(c1csc(=NCC)[nH]1)=O C1(CC)(CC)CC(NC(c2ccc(CO)c(F)c2)=O)CN1C(=O)C(C)N1CCC1 C1(C(=O)NCc2cc(C(=O)NCC(CC(C)C)OC)n(C)n2)CCN(OC)CC1 c1(C(=O)NC2CCC(CNC(CC(=O)OC)=O)CC2)cccc(=O)n1O C=CCC(C(=C)C)C(=O)N1CC2(CCN2C(=O)C=Cc2cccc(Cl)c2)C1 c1(C(N2CC3C(C(=O)NCc4ccccn4)C3C2)=O)cc(Br)nc(Br)c1 N1(C(C(=O)NCc2nc(C(C)OC)on2)=O)CCC(C(C(C)C)(OC)OC)CC1 O(NC(=O)C(C)N(C(=O)C=Cc1cc[nH]c1)CC)CC#C C(=O)(C(C)(C)C(O)C(C)C)NC(CCC=C)C(=O)N1CCOC(C#N)C1 c1(C(=O)NC(C)CNC(c2ccnc(C(F)F)c2)=O)cc(Cl)cc(F)c1N c1(C(=O)NC2C(NC(=O)CCN3CCOC3=O)CCOC2)cc2ncccc2s1 Cc1ccccc1C1(NC(=O)CN2CCN(Cc3nnc(C)s3)CC2)CCCC1 CCCCC(O)C(=O)NCC1CCC(NC(c2ccc(-c3cn[nH]c3)cc2)=O)C1 N1(C(c2cc(CCO)no2)C(=O)NC(c2ccccc2)C)CCSC(C)(C)C1 C(N=c1[nH]c(=NCC2CCCN2S(C)(=O)=O)[nH]c2c1SCC2)c1c(C)nccc1 O=C1CS(=O)(=O)CC(C(=O)NCC2COCCN2C(=O)COC2CCOCC2)N1 c1(C(N2CCC(N(C(=O)C(C)O)CCC)C2)=O)sc(-c2ccccc2F)nc1C C(=O)(C(CC(F)F)N(C(=O)CCP(C)(C)=O)C)NC(CC)(C)COC CC(C)CC(C(=O)N1CCSCC1C)ONC(C1(C)CNC(=O)C1)=O CCC(C(=O)N1CCOC(CN(C)C(C2CN3CCCC2C3)=O)C1)C(C)C c1(COC)ccc(F)c(C(=O)NC(c2csc(SC)n2)C)c1 N1(C(c2cc(C)n(CCO)n2)=O)CCC(NC(C2CCNC2=O)=O)C12CCC2 N12CCc3c(cccc31)C2.c1(CC)nn(C)cc1NC(=O)NC c1(C(=O)NC2C(c3cccc(NC(c4cn(C)nn4)=O)c3)C2)cc(Cl)ccc1Cl c1(CC(=O)N(CCOCCNC(C(CO)OC)=O)C)cccc(C)c1 c1(OCC(=O)NC(c2ccccc2)CNC(CC(C)C2CC2)=O)ccc(F)nc1 C1(CNC(COCC#C)=O)CCCN(c2cc(-c3ccc(C)s3)ncn2)C1 C1(C(=O)NCC2(CCNC(C3CC(n4cccn4)C3)=O)CC2)(OC)CC(C)C1 C1(N(C(=O)C=CCN2CCOCC2)CC)CCN(C(C2(C(C)=O)CC2)=O)CC1 N1(C(C2N(CC)C(=O)CC2)=O)CC23CCCC2(C1)CN(C(C1CC1C(C)C)=O)C3 N1(C(C2(CSC)CC2)=O)CCC(NC(=O)Cc2ccnn2C)CC1 N1(C(c2ccc(C#C)nc2)=O)CCCC12CCCN(C(=O)C(C)C(C)C)C2 CCCCC(CC)CC(=O)C(C=CCC(C)(C)NC(=O)N(CC)C(C)C)=O C(=O)(CCC(F)(F)C(F)(F)F)N1CCCN(C(CCN(CC)CC)=O)C(CO)C1 C(CCN(C(=O)Cc1cn(C)nc1Cl)C)(C(C)(C)C)NC(CC(CN(C)C)O)=O Cc1ccc(CN2CCOCC2C(=O)Nc2cnc(C)c(Br)c2)c(Cl)c1 c1(CC(N2CCCC(C(=O)O)C2)=O)ccc(C(F)(F)F)cc1Cl C1(CC(N2CC(CCCN)OCC2)=O)C2CC3CC(C2)CC1C3 CCC(CC)CC(=O)NCc1occc1C(=O)NC1CCOC1 C1(CC)CCN(C(=O)CONC(c2ccc(CC)c(F)c2)=O)CCO1 C(=O)(CC1=CCOCC1)N1CCC(O)(CN(C(COC(CC)C)=O)C)C1 Cc1ccc(C(=O)NC2(C(=O)NCCC3CCCC(C)C3)CC2(C)C)cc1 C1(Nc2c(C#N)cccc2)CCC2(CC1)CNC2 C1(C(N(C(C)C(N2CCC(F)C2)=O)CC)=O)CC(=O)CS1 c1(CN(C)Cc2ccc(C(=O)OC)o2)cccc(Cl)c1I CC1(C)CC(=O)N(CC(N2CC(CNC(=O)Cc3cscn3)C(O)C2)=O)C1=O CC1CCCC2(C1)NC(=O)C1(CC1)CN(c1ccccc1)C2.C(N)(=O)O.C(C#N)S c1(C(=O)NC2CCC(CNC(CSCCC)=O)CC2)csc2ccncc12 c1(OC(C)C)ccc(Br)cc1OC(c1cc(C(C)C)cc(Br)c1)=O c1(OC)cc(-c2ccc(C=O)s2)ccc1-c1nccn1C1CC1CC(C)CO C(=O)(CC(F)(F)CS(C)(=O)=O)N1CCC(CCc2cn(CCCC(=O)O)nn2)C1 N1(C(c2ncccc2O)=O)CCN(C(C2CCCCC2O)=O)C(C2CC2)C1 C(=O)(CC(CC)CC(F)(F)F)NC(CC#CC)C(=O)N1CCN(C)CC1 C12(CNC(COC(CNC(C3N(CCC)CCC3)=O)(C)C)=O)CCC(CC1O)C2 C1(C(=O)NCC(C)NC(c2ccc(Cl)cc2C(F)(F)F)=O)COCC2(CCC2)O1 n12cc3c(n1)C(N2)CCC3.C(=O)N=c1[nH]nc(-c2ccon2)s1.CCC N1(C(c2ccc(C)cc2Cl)=O)CCC2CN(C(=O)C(C)Cc3cnn(C)c3)CC12 Cc1ncc(C(N2CC3C(N(C)C(C4C5CC6C(C5)C46)=O)C3C2)=O)c(C2CC2)n1 C12(C(=O)NCCC3CC(NC(c4ccncc4Cl)=O)C3)CC3CC(C(=O)N1)C2C3 Cc1cccc2nc(C(N3CCC(NC(=O)CC(=O)NC4CC4)CC3C)=O)cn12 Cc1c(C(=O)NCC2CCN(C(C3CNC(=O)N3)=O)C2)sc2ccccc12 O=C(C1CCc2c[nH]nc21)NC1CCN(C(C23CCC(CC2F)C3)=O)CC1O c1(C(=O)NC2C(NC(Cc3ccn(CC)n3)=O)CCOC2)cc(C)cc(Cl)c1 N1(C(CSCC(N)=O)=O)CCC2CN(C(c3cccc4ncnn34)=O)CC12 c1(-c2c(C)onc2)cc(S(=O)(=O)Nc2ccccc2)ccc1C c1(C(=O)NC2C=CC(CNC(CCOC)=O)C2)cc(Cl)nnc1O.C1(N)CCCCC1 C1(NC(C2(C=C)CCCCC2)=O)CCN(C(c2cc(CC)no2)=O)CC(C)(C)C1 c1(CC)ccc(C(=O)NCC2COCC2NC(=O)C(F)(F)CC2CCCO2)nc1 n1(CCCC)ccc(C(=O)NCC2CCCN2CC)n1.C12CCC(C1)NC(=O)C2 C12(CCO)CCN(C1)C(=O)CSCCC(=O)N2.c1(S)cccc(Cl)c1.CC(=O)OCC c1(NC(CCN(C)C)=O)cccc(-n2cc(C3CCOC3)nn2)c1 C(=O)(C(F)CC(CC)CC)NC(CCCC=C)C(=O)N(C)CC1(C)CCCO1 N1(C(C=CCC)=O)CCC(C2CCN(C(=O)CS(=O)(=O)CC(C)C)C2)CC1 CCC(CC(=O)NCC(CO)NC(c1cnn(-c2ccccc2)n1)=O)C1CCC1 N1(C(=O)NCc2cc(-c3c(OC)cccc3)no2)CCCN(c2cccs2)CC1 c1(COC)cnc(N2CCC(NC(=O)C(C)NS(C)(=O)=O)CC2)nc1 C(=O)(C(C(C)C)C(C)C)NCC1CN(C(C2(SCC)CCCC2C)=O)C1 c1(C(=O)NCC2(Cn3cc(COC)nn3)COC2)nccc2[nH]nc(C(C)C)c12 N1(C(c2c(OC)csc2)=O)CCCCC1C1(NC(=O)CC23CC(C2)C(C)O3)CC1 C1(NC(c2ccc3nncn3c2)=O)CN(C(=O)CCc2ncc[nH]2)CC(F)(F)C1 CC1OC2CCC1(CNC(=O)C(n1cc(C3CCN(C)CC3)nn1)C)C2 C1(C(=O)NC2CC(CNC(=O)CN(C3CCCC3)C)C2)(OC(C)C)CCCC1 Cc1ccc2c(c1)C(=O)N(C(C)C(N1CC(C)(CNC(=O)C(C)CF)C1)=O)C2=O C1(C(=O)NCC2OCCN(C(CCc3cc(C)no3)=O)C2)CCCC12OCCO2 C1(N)CC(CN(C(CN(C(CN(C(C)=O)C)=O)C)=O)C)C1.C1(CO)CC1C c1(COC)ccc(-c2ccc(OC)cc2C(F)(F)F)cc1O N1(CC(C2CC2)OC)C2CCC1CC(NC(c1c[nH]c(C)cc1=O)=O)C2 C1(OC)CC(CNC(c2c[nH]nc2C)=O)N(C(=O)C=Cc2cscn2)C1 Cc1sc(Cl)nc1C(N1CCCCC1C(C)(C)CNC(=O)CC(C)(C)C)=O Cc1cnc(N2CCC(C3CCCCN3C(=O)C(C)(C)C)C2)nc1 N1(C(COCCOC)=O)CC2CC(NC(c3cccc(OC)c3OC)=O)CC1C2 Cc1cc(C)c(C(N2CCC2CNC(=O)C(F)CC2CCCC2)=O)[nH]1 CS(=O)C=CC(=O)NCCC1(O)CCN(C(=O)CCCSC(C)(C)C)C1 c1(CNC(C(C)SC)=O)ccc2c(c1)CN(C(C1CCC(C(N)=O)C1)=O)C2 c1(OC)cc(C(N2CCCCCC2CNC(=O)Cn2ccnn2)=O)c(F)c(Cl)c1 C12(NC(c3csc(C)c3N)=O)CCCN(C(c3cncc4nc[nH]c34)=O)CC1C2 N1(C(c2ccc(C)[nH]2)=O)CC2(CCN(C(=O)C(C)CC(N)=O)C2)C1 c1(CCCC)nc(C)c(-c2nc(C3CC3CC)nn2C2(C)CCS(=O)(=O)C2)c(O)n1 c1(COC)cccc(C(=O)NC2(C(=O)NC3(O)CCSC3)CC(C(=O)OC)C2)c1 C(C1CCCCC1)=C(C(N1C(CNC(C2CN(C(=O)NC)C2)=O)CC1)=O)F Cc1cc(C#N)cc(C(=O)NCC2CCCN2C(C2(C)CCC(C)CC2)=O)n1 CCCC(C(=O)NCC1CN(C(c2ccc(O)cc2N)=O)C1)C(C)C c1(C(N2C(CC)CCC2C(=O)NCc2cnccc2Cl)=O)cc(C)cc(C)c1 C1(NC(=O)Cn2nccn2)(CO)CCN(C(C2(Cl)CC2(F)F)=O)C1 N1(C(CC=CC=C)=O)CCC2(CCN(C(=O)C3CC3)CC2)C1 N1(C(c2ccc(C#C)cn2)=O)CC2CN(C(=O)C(C)(O)C=C)CCC12 C(C)(C)(C(C)CC(=O)N(C)C)NC(c1ccc(C)nc1C)=O C(c1ccccc1)=CC(N1C(C(C)NC(=O)C(O)Cc2cnn(C)c2)CCC1)=O c1(C(=O)NCCN(CCC)C(C2CC23CCCOC3)=O)ccc(F)c(Cl)c1F Cc1ccc(C(N2CCC(CCC(=O)N(C(CO)C3CC3)C)C2)=O)c(F)c1 c1(NC(Cc2c(NC(CC(CC)C)=O)cccc2)=O)cn(C)c(=O)nc1O C1(NC(CC2CC(OCC)C2)=O)CC2(CCN(C(C3CCC(F)CC3)=O)CC2)C1 c1(C2(C(N3CC(N(C(C(CC)F)=O)C)C3)=O)CCC2)c(F)cccc1F c1(C(=O)NCCCN(CCO)C(C2(F)CC2)=O)cccc([N+](=O)[O-])c1Br C=CC(O)C(=O)NC(C)(C(=O)NCC(F)Br)C1CCC1 C1(S(C)(=O)=O)(C(=O)NC2C(C)CN(C(C3(N(C)C)CCC3)=O)C2)CCCC1 c1(C(=O)NCC(CCOC)NC(=O)CC2CCOCC2)cnc(SC)n1C C(=O)(CC(C)CC(=O)NCC1CC(CNC(=O)CCc2ncc(C)[nH]2)C1)OC c1(C(=O)NC2CC(NC(CC3(C=C)CCC3)=O)C2)ccc(-c2cscn2)nc1 C(=O)(C1CCSc2ccccc21)NCC1N(C(CCCCC(C)C)=O)CCCC1 c1(OC)ccc(C(=O)NCCCCNC(=O)C(c2ccc(F)c(Cl)c2)O)c(F)n1 Cc1c(C(=O)NC(C)(CNC(=O)CCc2cccs2)Cn2cccn2)cccc1N Cc1ccc(C(O)C(=O)NCCC(O)CNC(=O)CN2CCC2C)cc1 Nc1ccc(Cl)cc1C(=O)NCCNC(c1cnc(Br)s1)=O CCS(=O)(=O)C1CC1.C(C(=O)NCCO)N.C(=O)(CS)N(CCCCSC(F)F)C C12(C(=O)NCCCCCCNC(c3n(C)cnc3)=O)CCOC1CS(=O)(=O)C2 C1(C)(C(=O)NCC(C)NC(=O)CC2CCC(=O)NC2=O)CCN(C)CC1 CC(O)C(C(=O)N1CCC(N(C)C(C2(F)CCCC2)=O)C1)N(C)C Cc1ccc(C(N2CCCC2C2(NC(=O)CN3CCC3C)CC2)=O)c(Cl)c1 C1(O)(CC(N2CCC(C(C)NC(=O)COC3CCOC3)CC2)=O)COC(C)(C)C1 c1(C(C(=O)OC(=O)C(O)CC2CCCCC2)OC(CC=C)C)cccc(C(F)(F)F)c1 CC(CC(=O)N(C)CCN(C(=O)CN(C)CCO)C)C1CCCO1 N1(C(C=CC2N(C)CCC2)=O)CCC(C)(C)C1CC(=O)NCCCN1CCCC1 C12(C(N(C(C)C)CCN(C(=O)C=CC3CC3)C)=O)CCCN(CC1)C2 Cc1ccc2c(NC(N3C4CN(Cc5cc(F)ccc5Br)CC34)=O)cccc2c1 c1(OC)cncc(Br)c1C(=O)N(C)CCOCCN(C)Cc1cnsn1 C1(CF)CCCN(c2ccnc(N3CC(NC(C4CCC4)=O)C3)n2)C1 CN1CCOCC1C(N1CCC(C(C)(C)C(N2CC(O)CC2C2CC2)=O)C1)=O N1(c2ccnc(OC)n2)CCc2ccc(C(=O)Nc3ccc(Br)nc3Cl)cc2C1 c1(C(=O)NCC2(O)CCN(C(CC3NC(=O)OC3)=O)C2)cccc([N+](=O)[O-])c1 C1(CC)(CO)CCN(C(C2CC3CC3N2C(=O)CC23CCCC2C3)=O)C1 c1(C(N(C(C)C(=O)NCC2CC(C#N)C2)CCC)=O)c[nH]c(=O)cn1 C(CCC(=O)N1CC(C2CC2(F)F)C1)(C(C)C)NC(c1cc(=NC)[nH]cc1)=O C1(NC(CSCCOC)=O)CC2CN(C(c3cc4sc(C)cc4s3)=O)CC2C1 c1(CC)nn[nH]c1C(N1CC(CCCCNC(=O)CC2CCC3CC23)C1)=O N1(C(c2ccc(CC)[nH]2)=O)CC2(CCC(NC(C3CC(C)C3)=O)CC2)C1 CN1CCN(C(C2(C)CCNC2=O)=O)CC1C(=O)NCCNC(=O)C1CC1 N1(C(C2(CC#C)CC2)=O)CCC(C)(C)C(C(N2CC=C(C)C2)=O)C1 N1(C(CNC(C2CC23CC3(F)F)=O)=O)CCN(C(=O)COCCC#C)CC1 c1(C(C(N2CCN(C(C3CSC3)=O)CC2)=O)OC)cccc(-c2cn[nH]c2)c1 C#CC1(C(N2CCC3CC23)=O)CCN(C(=O)Cn2cccc2)C1 c1(NC(N2CCC(c3ocnc3Br)C2)=O)ccnn1-c1cn[nH]c1 C1(CC(=O)N(CCSC)CC)CCCCCN1C(C1CCC(O)CN1C)=O C=C1CC2CC1CC2(c1nnnn1Cc1cc(Cl)ccn1)NCC12CC(CCO1)C2 C1(CC=C)(C(N2CCC(O)(C(F)F)C2)=O)CCCN1C(=O)Cc1ccc(C)s1 C1(N(C(C(CC)N(C)C)=O)C)CCCN(C(=O)CCCC2CCC2)CC1 C1(NC(c2cc(CC)[nH]n2)=O)CN(C(=O)C(O)C(C)(C)C)CC1N=[N+]=[N-] N1(C(c2c(C#C)cn(C)n2)=O)CCC(C)N(C(c2cn(CC(N)=O)nn2)=O)CC1 Cc1cc(=NCCCNC2CCCCC2)[nH]c(=NCCC(C)N(C)C)[nH]1 N1(C(Cc2n[nH]c(=NC)s2)=O)CCC2CCCC(C1)N2C(C1(C)CC2CC2C1)=O C(CC(C(C)(C)C)NC(=O)C(C(C)(C)C)SCCN)N(C(CCC(=C)C)=O)C C1(NC(C2C(C(=O)OC)C2)=O)CC(C(=O)N(C)Cc2cnn[nH]2)=CC1O Cc1ccnc2nc(C(N3CC4(CCN(C(C5(C)CSC5)=O)C4)C3)=O)nn12 c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(C)(C)C)c[nH]c2ccc(C)cc12 c1(CC(=O)NC2(CN(C(=O)CC3CC3)C)CC2)csc(N(c2ccccc2)C)n1 c1(C(CNC(c2cn(C)nc2)=O)NC(C2CCC3CC23)=O)cccc(Cl)c1Cl CC1CC(C(=O)NC(C)(CNC(C2CCSC(C)C2)=O)C2CC2)=NO1 N1(C(CSC)=O)CCCC1CCNC(c1ccnn1C1CC1(F)F)=O c1(NCC2CCC(C(=O)O)CC2)ccc2c(c1Cl)CCC2=O C(=O)(C(CC)C(=O)NC(C(N1Cc2c[nH]nc2C1)=O)C(C)C)OCC N1(C(C(CC)C#N)=O)CCOC2(CCCN(C(c3cnn(C)c3SC)=O)C2)C1 C1(C)(C(=O)NCCC(C)C)CC(O)CN1C(=O)CC1CSC1 c1(NCC2C(C)CN(C(c3cc(Cl)c(Cl)[nH]3)=O)CC2)nc2c(cc1Cl)C(=O)OC2 N1(C(CCOC(C)C)=O)CCC2(CC1)CN(C(C1CC1(Cl)Cl)=O)CC(C)O2 C1(NC(c2cc(CC(C)C)on2)=O)CC2CC1CN(C(=O)CC1CCN(C)C1)C2 c1(CCC(=O)NC2C(NC(C3C(=C)C3)=O)COC2)ccc(Cl)cc1Br c1(C(CNC(CC2CC(OC)C2)=O)NC(=O)CCCn2cccn2)ccc(F)cc1 N1(C(CCC(C)=O)=O)CC(C(N2CCCC(CO)C2)=O)C(C2CC2)C1 N1(C(c2ccn(CC)n2)=O)CC(C)CCC1CNC(=O)C(C)(C)C(N)=O CC1=C(C(=O)NC(C(=O)NC(C)CO)C2CCCC2)COCC1 Cc1cc(C(=O)NCC2CC(C(=O)NC3(CO)CCOC3)C2)c(N)s1 C1(CN(C(CC(=C)Br)=O)C)CCCN(C(=O)Cc2cnco2)C1 C1(N(C(C2CC2c2ccoc2)=O)CC)CC2(CCC2)CN1C(=O)C=CC(C)(C)C C1(C(N2C(CNC(c3ccc(NC)cc3)=O)CCC2)=O)CCCC1C1CC1 c1(C(N(CCCNC(=O)C(C)C2CCOC2)C(C)C)=O)cnc2scnc2c1 c1(C(C)NC(c2cc(Br)ccc2Br)C)ccc2c(c1)OC(F)(F)O2 C1(CC(=O)O)CN1.C(C)(C(=O)N(C)CC1CC1)SCC Cc1nn(C2CCC2)cc1C(=O)NCC1(F)CCN(C(c2sccc2F)=O)C1 C=C(C)C1OCCC1C(=O)NCc1cc(C(=O)N2CC(O)CO2)cs1 C1(CNC(C(C)OCC(F)(F)F)=O)CN(C(=O)C(c2cccnc2)C)CCCO1 C(=O)(C#CC1CC1)NCC(CCNC(CC=CC=C)=O)O C1(C(=O)OCC)CN(C(c2cc(Br)ccn2)=O)CC12CCNCC2 C1(C(C)(C)CNC(C2CC=CCC2)=O)CCN(C(c2csc(C(F)F)c2)=O)CC1 C(C(CC(=O)NCCC(C)N(C)C1CC1)C1CCC1)NC(COCC)=O c1(C(N2C(CN(C(C3C(C)=C3)=O)C)CCC2)=O)ccc2scc(C)c2c1 C(CCC(=O)N1CCC(CN(C)C)C1)N(C(C=C(COC)C)=O)C N1(C(C2(C)CCOCC2)=O)C2CCC1CC(CNC(C1C3CCCC13)=O)C2 N1(C(c2n(COC)ncc2)C(=O)NCCC2CC2)CCC(CSC)C(O)C1 c1(SCC(=O)NC2CC(NC(C(C)OCC(F)(F)F)=O)C2)cccc[n+]1[O-] N1(C(C(C)OC2CCOCC2)=O)CCC2(C1)CN(C(c1nccn1C)=O)CCO2 C(CC(C(=O)NCC1=CCCCC1)NC(=O)CC1CCCC1)OCC c1(OCC(=O)NC(C)CNC(=O)CN2CC3CC3C2)cc(F)cc(F)c1 c1(C(N2CC(NC(CCC(=C)Cl)=O)C(O)CC2)=O)ccc2c(c1)OCO2 CC1=C(C(=O)NC2(C)CC(NC(C3CCN(C)CC3)=O)C2)Cn2ncnc2N1C c1(C(=O)NC2CCCCN(C(CCCC#N)=O)C2)c(Cl)oc2ccccc12 S(=O)(=O)(c1cnn2ccc(N3CC4CCC(F)(F)C4C3)nc12)NCc1n(C)cnc1 CC1CCc2nc(C(=O)NCCOCCN(C(=O)C(C(C)O)N(C)C)C)cn2C1 CCC(O)C(C)C(=O)N(C1CCN(C(=O)CSCc2ccc(C(N)=O)cc2)C1)C C1(NC(CCC2(C)CN(C(=O)C=CCF)C2)=O)CCOCC12CCC2 CCC(CC)(CC)C(=O)NCCn1cnc(C(N2CCOCC2)=O)c1 CC1OCCN(C(c2cnc(Cl)n2C)=O)C1C(=O)NCc1ccc(O)c(F)c1 C#CCC(C(=O)NCC(C)(CC)CC)NC(=O)Cn1nnc(C)n1 N1(C(c2c(COC)scc2)=O)CC2CN(C(=O)C(c3ccccc3C)C)CC2C1 N1(c2ccnc(C(C)C)n2)CCC2CC(C(N3CCCC(CO)C3)=O)C2C1 C1(CNC(C(CC)(C)OC)=O)CC2CCCC2N1C(c1ccnc(C(F)F)c1)=O Cc1cc(C#N)cnc1C(N1CCCOC(C(=O)NC2CCOC2)C1)=O CS(=O)(=O)CCCC(=O)NCCCCCCNC(c1nc(C2CC2)cs1)=O c1(C(N(CCC)CCNC(C2CC2(F)Cl)=O)=O)cn(C(C)(C)C)nc1C(C)(C)C C1(CCNC(=O)CCC2CCCC2)CCC(NC(C2(n3cncn3)CC2)=O)C1 C=CCC(C(=O)NC1CCC(NC(C2CCCC(CF)C2)=O)CC1)NC(C)=O C#CC1(C(=O)NCC(C)=CC(=O)NC2CC3(C2)CC3(F)F)CCCCC1 N1(C(=O)OCC)CCC(C(C)NC(=O)C(=O)NCC2(C)CSCCO2)CC1 c1(CN2C(C(=O)NCc3cccc(OC)c3C)C=CC2)ccc(O)c(C)c1O c1(C(N(CCNC(=O)Cc2ccc(OC)cc2)CC)=O)cc2cccc(Cl)c2[nH]1 C#CCC(C)(C(=O)NC(CO)CCC(C)C)NC(c1occ2c1CCC2)=O c1(C(=O)NCCN(C(C2(CC)CNC(=O)C2)=O)CC)cccn2cncc12 C1(C(N2C(C)(CCC)CC2)=O)CN(C(=O)OC(c2ccccc2)CC)CCO1 N1(C(COC(C)=O)=O)CC2CC(NC(c3ccccn3)=O)CC(C2)C1 n1(C(C)C)cnc2c(N3CCOc4ncccc4C3)nc(N(C)C)nc12 n1(CCCOC)nc(-c2cccc(SC3CCC3)c2)nc1-c1cocc1C c1(OCCCC)ccc(NC(=O)CCOc2ccccc2)cc1.C1(=O)CO1 N1(C(CNC(=O)OCC)=O)CCC(NC(c2cccnc2C)=O)CC1C1CC1 C1(CNC(c2cnc(C)o2)=O)CC(C(=O)NC2CCC(C)(C)CC2)=NO1 c1(-c2cc(C(N(CCCNC(c3cnc(SC)s3)=O)C)=O)no2)ccccc1C c1(C=O)ccc(CC)cc1.N1(C(CC=C)=O)CCCC1 CCC(O)C(C)C(=O)NCCN1CCC(NC(=O)Cn2cc(F)ccc2=O)CC1 NC1CCCC(C(=O)Nc2ccc(F)c(Sc3ccccc3)c2)CC1 N1(C(c2c(N)ccc(C(C)C)c2)=O)CCCN(C(C2CC23CC3)=O)C(C)C1 Cn1c(O)ncc(CC(N2CCC2Cc2ccc(Br)cc2)=O)c1=O C(N=c1ccc(Br)c(S(=O)(=O)N)[nH]1)C1C(C)(C)C1.n1(C(N2CCC2)=O)cc(CO)cn1 N1(C(C(CCC)OC)=O)CCC2(CCCN(C(C3(c4ccsc4)CC3)=O)C2)C1 CON(CCC(=O)N1CC2(CCCCO2)C1)C(=O)CCCC1CC1C N(C(=NCC1CCOC1)NCC1(CO)CCOCC1)C(C)C CCCC(C)CC(=O)N1CCCC1CN(C)C(c1ccc(CSC(F)F)o1)=O C1(NC(C(C)OCC#C)=O)CC2(C1)CC2C(=O)N(CC(F)F)C1CC1 O=C(CC1CC2CCCC2O1)N=c1ccn(CCOC2CC3(C2)CC3(F)F)[nH]1 Cc1cnn2c1CN(C(c1n[nH]c3c1CN(C(C1CCC(F)C1)=O)C3)=O)CC2 N1(C(C2CCCC(OC)C2)=O)CCC(O)(CN(C)C(C2COC2)=O)CC1 CC(C)C(O)CC(=O)N1CCCOC(CNC(=O)CCc2ccccc2)C1 C1(C(N2CC(SC)C2)=O)(NC(CN(CC)CC)=O)CCOCC1 c1(OC)ccc(F)cc1C(N1CCC(CF)(NC(=O)CC(C)C(C)C)C1)=O c1(C(N2C(C)(CC(N3CC(CO)CC3CO)=O)CC2)=O)cc(C#N)cs1 c1(CN(C(C(=O)NC(n2cc(Br)cn2)CF)=O)C2CC2)ccc2ccccc2c1 c1(CCNCc2cc[nH]n2)cccc(F)c1OC(F)(F)F.C12CN(CCO1)C2=O CON1CC(C(=O)NCC(C)(O)CNC(c2nc(C)no2)=O)CC1=O C(C(=O)OCC1CC1)(C(C)C)NC(CC(=O)NCCCOCC)=O CC(CCCNC(=O)C(=O)N1CCC1c1ccccc1)NC(C1CC(O)C1)=O c1(C(=O)NN2CCC(N(C(c3c(CC)nn[nH]3)=O)C)C2)cnc2n1CCS2 C(O)(CC(=O)NC1CCCCN(C(=O)CCCC(F)(F)F)C1)(C(F)(F)F)c1cn(C)nc1 N1(C(CCC(=O)NCCC)=O)CCCC(NC(C2(C)CC3(CCC3)C2)=O)CC1 C1(NC(c2ccc(OCC)nc2)=O)CN(C(=O)CC2OCCO2)CCC1C CC(C)C(O)C(C)(C)CN=c1[nH]c(=NCCS(=O)(=O)NC2CC2)c2cc(Cl)ccc2[nH]1 c1(NC(C2(F)CCN(C(C(OC)OC)=O)C2)=O)cc(C)c(F)c(C)c1 CCC(C)(C)C(=O)C(=O)NCC1CCCCN1C(=O)C(C)OC1CCCCCC1 c1(C(N2CCC(C(C)NC(C(CC3CCC3)OC)=O)CC2)=O)ccnc(C)c1N C1(NC(CNC(c2ccc(C)cc2)=O)=O)CCCCN(C(C2(CO)COC2)=O)C1 Cc1c(Cl)cnc(NC(C)CCNC(=O)C2=NOC(C(C)(C)C)C2)c1C#N C1(C(N2CC(C)(NC(=O)CCn3cccnc3=O)C2)=O)CC12CC(F)(F)C2 C(=O)(C1=CC2(CCOC2)C1)N1CC(NC(=O)C(CO)C(F)(F)F)C2(CC1)CC2 C1(c2nnnn2C2CCCC2)(NCC2(OC(C)C)COC2)CC(C(C)(C)C)C1 C1(CNC(C2(CCC=C)CC2)=O)CC2CCC(C1)N2C(c1cccc(F)c1F)=O N1(C(C2CCC(CC)C2)C(=O)NCCN2CCOCC2C)CC2(CC2)CC1C CCS(=O)(=O)C=CC(=O)N1CCCC1c1cn(Cc2nonc2C)nn1 CC1CC(CNC(c2cc(Cn3cccn3)on2)=O)CN1C(=O)C(F)F Cc1csc2c(N3CC4CCC3CN4Cc3ccc(F)cc3)ncnc12 O=C(C1CCCc2ccccc21)NC1CC2CCC1N(C(C1CC1C1CC1)=O)C2 C1(C(N(CCNC(=O)C2=CCCC2)CCOCCO)=O)CC2CC(=O)C1O2 c1(-c2onc(C(C)C)n2)ccc(C=CCC(=O)NC(C)CC2CC(CF)C2)cc1 c1(C(N2CCC(C)C2CNC(c2cc(=O)cc[nH]2)=O)=O)cc(O)ccc1O N1(C(CS(=O)(=O)N(C)C)=O)C(CNC(c2cnc[nH]c2=O)=O)CC2CC12 N1(C(C(C)OCC)=O)CC(C)C(C)(CNC(C2CN3CCC2CC3)=O)C1 c1(C(N(CCC(N2CCC(OCCF)C2)=O)CC)=O)nnccc1C O=C1NC(=O)C2(CCCC2CNC2CCN(c3ccc(F)c(Cl)c3)C2=O)N1 c1(C(=O)NC2C(OC)CN(C(c3ccc(F)c(C#N)c3)=O)C2)cc2scc(C)c2[nH]1 C=CCC(CC=C)C(=O)N1CC2(CCCC2NC(=O)C(O)Cc2cnn(C)c2)C1 c1(C(=O)NCC2N(C(C(CO)N(C)C)=O)C3CCC2C3)ccc([N+](=O)[O-])cn1 C(C(C(=O)NC1CCCCNC1=O)C(C)(C)C)NC(c1c(OC)ccnc1)=O c1(C(N2C(C(=O)OCC)C=CCC2)=O)[nH]c(C)c(C(C)=O)c1C C1(C(=O)NC23C(CN(C(c4n[nH]c(CC)c4Cl)=O)C2)C3)CC12CCS(=O)(=O)CC2 N1(C(c2[nH]cc(C(N)=O)c2)=O)CC2CC2C1CNC(C1CCC(C(N)=O)CC1)=O N1(C(c2nn(CC)c(C(F)(F)F)c2)=O)CCOc2ccc(C(=O)NC)cc2C1 Cc1ccc2c(Cl)c(C(N3CCC(CN(C(=O)C(C)CF)C)CC3)=O)sc2c1 c1(C(C)(F)F)ccc(F)c(C(=O)NC2CC(Cn3cc(-c4nccs4)nn3)C2)c1 C1(C2CC2)(COC)CN(C(c2conc2C(C)NC(=O)C(C)C2CCCC2)=O)C1 Cn1ncc2ccc(C(=O)NC3C4CC3N(C(C3(C)CCCCC3)=O)C4)cc12 CC(CS(C)=O)C(=O)N1CC(C(N2CCC(N3CCCCC3)C2)=O)C1 CC1C(C)N(C(c2ccc(C#N)s2)=O)CCN1C(=O)CCCC(F)(F)F N1(C(C(C)(O)C2CC2)=O)CCCC2(NC(=O)C(C3CCOCC3)O)CCCC12 CS(=O)(=O)C(CNC(=O)CN1CCCCC1)CNC(C1CCCN1C1CC1)=O CCC(C)CC(C)N(C)C(c1ccoc1CNC(c1cnn(CCO)c1)=O)=O Cc1cncc(C=CC(=O)NC2CC2NC(c2coc3c2COC3)=O)c1 c12ccc(Cl)nc1NC2=O.C1(CC(N)=O)COCCN1C(c1cccc(Br)c1)=O N1(C(c2cc(CNC(c3ccc(C(F)(F)F)s3)=O)on2)=O)CCCC(O)(CO)C1 C1(CCN2CC(c3ccccc3)(NC(c3cccc(Cl)c3)C)C2)CCC(C)(C)O1 C1(CNC(=O)C(F)F)CN(Cc2ncnn2-c2cccc(F)c2)CCO1 CC(C)CC(C)(CNC(c1cc(N)cc(O)c1)=O)NC(=O)CC1CC2CCC1O2 c1(C(N2CC(NC(C3CCCS3)=O)CC(C)(C)C2)=O)ccc(Cl)c2occc12 N1(C(C2(C)CCC(C)CC2)=O)CCOCC(C)(CNC(=O)COC(F)(F)F)C1 C1(CCC)(NC(=O)C(C)OC)CCCN(C(c2ccc(N)cc2OC)=O)C1 c1(C(=O)NC2CCCC(NC(C3C(CN(C)C)C3)=O)C2)c(F)ccc(F)c1O C1(CN(C(CCC2C(C)C2)=O)C)C2CN(C(=O)CCCc3cccs3)CC12 C1(SC)CC(c2nc(-c3ccc(I)cc3)nn2C2CCCC2)CCO1 c1(C(N2CC(C)(NC(=O)C=CCN3CCCCC3)C2)=O)ncc(Cl)cc1F c1(S)ccc(F)cc1.CC(O)(C(=O)NC1CC(C)(NC(=O)CC2CC3(CC3)C2)C1)C1CC1 C(=O)(CCSC(C)=O)NCCN(C1(C(=O)NC)CC1)C(C)=O.OC c1(C(=O)NC(C(=O)NC(C)Cn2ccnc2)Cn2ccnn2)cn(C)cc1C C12(C(=O)NCCCn3cc(-c4ccccc4)nn3)CC3CC(C(=O)N1)C2C3 N1(C(c2c(C)nc[nH]2)=O)CCC2(CCCCC2NC(c2csc(CO)n2)=O)C1 Cc1cc(=NC2CCCc3c[nH]nc32)[nH]c(=NCc2cc(Cl)nc(=N)[nH]2)[nH]1 C1(C)(C(N2C(C(=O)NC(CC(C)C)CO)CC2C)=O)CC2(CCC2)C1 c1(C(=O)NCCN(CCC)C(C2(C#N)CCOCC2)=O)ccc(OC)cc1C C1(O)(CC(=O)NCCN2CCCC2=O)CCN(C(C2(CC3CCC3)CC2)=O)C1 CCCCC(C)CCC(=O)NCC(=O)NCC(=O)N(CC(C)(C)O)C CCC(O)C[SH](C)(=O)NNC(=O)c1cc(Br)ccc1F C(CC(C)C)(C(=O)NCc1ccc(N)cc1)N(C(C(C)(C)OCCC)=O)C CC1c2ccccc2OC1CC(=O)NCC12CCCC(CN1C(=O)CNC=O)C2 C#Cc1ccnc(C(=O)NC2CCCCC2NC(=O)CCNC(=O)CO)c1 C(C)(CC(C)(C)OC)NC(C(C)N(C(C(C)=C(CC)C)=O)CC1CC1)=O N1(C(C2N(C(C3CC(OC)C3)=O)CCOC2C)=O)CCn2c(C)cnc2C1 c1(OC)ccc2occ(C(=O)NCC(C3CC3)NC(C3ON=C(C)C3C)=O)c2c1 C1(NC(CCCn2c(C)cc(C)n2)=O)CCCN(C(c2ccsn2)=O)C1C C1(CC)CN(C(=O)CC2(C)CCCO2)CCN1C(=O)CCOc1cccnc1 c1(CC)ccc(C(=O)NCC23CC(NC(c4c(C)nsc4N)=O)(C2)C3)nc1 C1(C(=O)NCC(C(C)(C)O)O)CC(O)CCN1C(=O)C=Cc1cc[nH]c1 C1(C(N(C(C)(C)C)CCO)=O)C2CCN(C(=O)Cn3nccn3)CC12 c1(C(=O)NC2CCN(c3c(OC)ccc(Cl)c3)C2)cc(S(N)(=O)=O)c(Cl)o1 C(=O)(C(OC)OC)NC1CCOC1.C1(=O)CN1CCOC CC1=CCC(C(N2CC(O)(C(=O)NC(c3cnn(C)c3)CO)C2)=O)CC1 c1(C(=O)NCC(=O)NC2C(C)CCC2)n[nH]c2c1CS(=O)(=O)CC2 C=CCC(C)N=c1[nH]c2c(c(=NCc3ncc(Br)s3)[nH]1)CC(C)CC2 C1(CNC(c2onc(CC)c2C)=O)CCN(C(c2[nH]c(C)nc2C)=O)CC1(F)F C(=O)(CCCCC(=O)NCCC1CN(C(=O)C(C)(F)C(F)(F)F)C1)NC c1(OC)ccc(N2CCC3CC3C2)cc1NCCC1CC(=O)N(C)C1 N1(C(C2N(C)C(=O)NC2)=O)CCC2(CCCN(C(c3cnncc3O)=O)C2)C1 C(C)(C(=O)NN=c1[nH]ccnc1F)c1ccc(C)o1 CC1CN(C(c2cc(C(N)=O)co2)=O)CCC1CNC(=O)C(C)(C)c1ccsc1 C(CC(O)C(=O)NCC(C)N(C)C(C1CCCC1(C)C)=O)SC C1(C(C)C)C(=O)N(C)CCN1C(c1cc(Br)ccc1F)C(=O)NCC1CCCO1 N1(C(c2c(CC)c(C)ccc2)=O)CCC2(CC(NC(C3(C)CCCN3C)=O)C2)C1 c1(CC(N2CCC(N(C(C3CC(N(C)CC)C3)=O)CC)C2)=O)ccc(F)c(C)c1 c1(C(N2CCC(F)(CNC(C(C)n3cccc3)=O)CC2)=O)ncsc1S(N)(=O)=O c1(CNC2CCC(NC(c3csc(Cl)n3)=O)C2)cc(F)ccc1Br c1(C(=O)NCc2ccc(CNC(C34CC(F)C3C4)=O)cc2)ccc2nonc2c1 C1(NC(CN2CCN(C(c3nc(C)c(C)s3)=O)CC2)=O)CCCC(F)(F)C1 C=CC(CCC)CC(=O)N1CCCC1(C(=O)NCCc1nccn1C)C(C)C S(=O)(=O)(c1cccc(C(=O)NC2CC2CNC(=O)C#CC(C)(C)O)c1)NCC#C c1(C(C)C)ccc(F)c(C(=O)NCC(C2CCOC2)NC(=O)CNS(C)(=O)=O)c1 c1(C(=O)NCC2CCN(C(=O)COC3CCCC3)C2)cc2ccccc2o1 c1(C(=O)NC2C(CNC(c3ccc(Cl)cn3)=O)CC2)cc2ccncc2s1 C1(NC(CCCC=C)=O)CCC2CCN(C(=O)CSc3nccn3C)C12 CC(C)CC(C(=O)N1CC(=O)NC(C(C)C)C1)ONC(c1nccn1C)=O c1(N2CCC(CNC(N(CCOC)C(C)C)=O)C2)cc(C)c2[nH]ccc2c1 C(=O)(CCC1=CCCCC1)N(C1CCN(C(CCCCC=C)=O)C1)CC1CC1 C(=O)(C#CC1CCCOC1)NCC1(C)N(C(Cc2cc(C)no2)=O)CC(F)(F)C1 CC12CCC(C(=O)NCCC3CN(C(=O)C=Cc4cncs4)C3)(CO1)C2 c1(C(=O)NC2CN(Cc3cccc(C(F)(F)F)c3)C2)ccnc(Br)c1 c1(CC(=O)N(CCC(C)NC(=O)CCc2cn(C)cn2)C)csc2nccn12 C1(O)(CNC(c2c(C(C)NC(C3CC4CC4C3)=O)noc2)=O)CCCC1(C)C c1(CC(=O)N(CC)CC2CC2(C)C)csc(CNC2CCN(C(C)(C)C)C2)n1 C(C1CCc2ncnn21)NC1(CNC(C2C(CC)C2)=O)CCOCC1 Cc1ccc(C(=O)NCC(C)NC(c2cc(C(N)=O)c[nH]2)=O)c(F)c1Cl CCCCC(CC)CC(=O)NCc1nocc1C(=O)N(CC(C)C(C)C)C c1(C(=O)NCCC2(O)CCN(C(C=C(COC)C)=O)C2)ccc(Cl)c(Cl)c1 n1(CC(NC2=NCCN(CC=C(C)C)C(=O)N2)=O)nc2ccccn2c1=O C1(C(=O)NCC2(CCC)CCC2)CCN(C(C)=O)C(C)(C)C1.C12CN(C1)C2=O C1(C(N2CC(c3cn(CCC=C=C)nn3)(C)C2)=O)CCC2(CCOCC2)O1 C1(OC)CCC(CC(=O)NCC2(C)CC(C(=O)NC3COCCOC3)C2)CC1 N1(C(C=NOC)=O)CCC(CC(=O)NOCC2(C)CCC2)C1(C)C C1(NC(C23OC(C)C(C2)C3)=O)CCN(C(=O)C(F)(F)c2ccccc2)CC(O)C1 N1(C(C2CCC(N(C)C)CC2)=O)CC2=C(C1)CN(C(c1ccc(Cl)cc1N)=O)C2 c1(-c2nc(C)c(C(=O)Nc3cc(Cl)cc(I)c3)cc2)c(F)c(F)c(O)c(F)c1F N1(C(CC(C(C)C)C)=O)CC2CCCC(Nc3cc(Cl)ncn3)C2C1 c1(CN(C(=O)C=C2CC2)CCNC(C(n2cc(Cl)cn2)C)=O)cccc(Cl)c1 CC1CN(C(=O)Cc2ccc(Cl)s2)CCCN1C(c1cc(C#N)ccc1O)=O C1(C(=O)Nc2nccc(C(F)F)n2)CCCNC1c1ccccc1 N1(C(C(C=C=C)C)=O)CCN(C(=O)Cc2c(Cl)cnn2C)CCC1C N1(C(CCC=C(C)C)=O)CC(CNC(=O)OC(C)(C)C)CC1C1CCCC1 c1(OC)ccc([N+](=O)[O-])c(N(C)Cc2ccccc2CNC(=O)C=CBr)n1 N1(C(c2c(N)cc(F)cc2)=O)CC2(C1)SCCC2NC(C1CC12CCCC2)=O C=Cn1nccc1C(=O)N(CC(C)(C)NC(=O)C(C(C)C)NC(=O)NC)C C1(NC(=O)C(c2ccccc2)F)CCCCN(C(C2(Cl)CC2)=O)C1 c1(C(=O)NCCOc2c(C)cc(I)cc2)cc(F)c(F)c(Cl)c1 Cc1cc([N+](=O)[O-])ccc1-n1cc(C2CCCC2NC(c2n[nH]cc2Br)=O)nn1 C(=O)(C(C)C(C)(C)C)NCC1(NC(C(c2ccc(F)cc2)OC)=O)CCC1 N1(CC(=O)NC2C(NC(C3(C#N)CC3)=O)CCC2)CC2CCC1C2 c1(OC)ccc(C(N2CCCC(N(C)C(C3CC4CCC3N4)=O)C2)=O)cc1F N1(C(C2CC(=C)C2)=O)CCC(CNC(C2(CCc3ccccc3)CC2)=O)C1 C1(COC)(NC(=O)Cc2nnc(C)s2)CCCN(C(=O)C(C)(C)C(C)C)C1 N1(C(c2ccc(C)cn2)=O)CCN(C(=O)C(C)Cc2ccccc2)C(C)C1 c1(OC)cccc(CC(C)CC(=O)N2CCC(NC(c3cc(OC)no3)=O)C2)c1 n1(CC)ccc(C(=O)NC2COCC2CNC(=O)C(C)=CC(C)(C)C)c1C CC1=C(C(=O)N2CC3CC(C(N4CC(O)CCC4C)=O)(C3)C2)CCO1 C1(CC(=O)NCCC(CNC(c2cnc(C(C)=O)s2)=O)O)CCCNC(=O)C1 CC(C)C(O)CC(=O)N1CCC(F)(CNC(=O)COCC2CC2)C1 CN1CCC(n2nc(Cc3cnsc3)nc2-c2ccccc2)CC1 Cc1nccnc1C(=O)N(CCC(=O)NC1CCCC(C)C1)C1CC1 CC(O)CCCC(=O)N1CCN(c2cc(C(=O)NC3CC34CCC4)ccn2)CC1 C1(c2nccc(OCC)n2)CC(OC)CCN1C(=O)C=Cc1cccc(O)c1 CN1CC=C(C(=O)NCC2(NC(=O)COc3ccccc3F)CCCC2)C1 C1(NC(C(C)OCCN(C)C)=O)CCC(N(C)C(c2ccnnc2)=O)CC1 c1(NC(C2CC(NC(C3CC(=O)NC3)=O)C2)=O)ccc(C(F)F)c(F)c1 n1(CC(=O)NC2C(CC)CN(C(=O)CC3CCSC3)C2)ccc(=O)cc1C N1(C(c2nc(C)[nH]n2)=O)CC(C)CCC1CNC(c1cc(C)c(C(F)F)cn1)=O C12(C(=O)NC(C(C)C)(C)CNC(c3ccc(C#N)cn3)=O)CCCN(CCC1)C2 C1(NC(C2(C)N(C(C(C)C3CCCC3)=O)CC=C2)=O)CCCCCC1C N1(C(C2ON=C(C)C2C)=O)CCN(C(C2CC(O)C2)=O)CC12CC2 c1(C(N(C(C)CCNC(=O)CN(C)C)C)=O)cc(C(F)(F)F)ncn1 C(N=c1cccc(S(=O)(=O)NCC(CO)CO)[nH]1)c1c(N)cncc1 Nc1cc(C(=O)NCC2CN3CCN2CC3)cc(Br)n1 CC(C)CCCC(=O)N1CC2CC1C2C(N1CCC=C(F)C1)=O c1(C(=O)NCC(CO)NC(C=Cc2c(C)nccc2)=O)cc2c([nH]1)CCCC2=O CCCCCC(C)CC(=O)NC1(C)CN(C(C2CCn3nc(C)nc3C2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)C2CCC1CC(CNC(C1(F)CCCOC1)=O)C2 C(=O)(C1=C(C#N)CCC1)N(CCC(N1CCC(CN(C)C)C1)=O)CCCO C(=O)(CC(C)CC(=O)NC(C)Cn1cc(-c2cscn2)nn1)OC Cc1oc(C#N)cc1C(N1CC(C(=O)NCCC2(CO)CC2)CCC1C)=O S(=O)(=O)(c1ccc(C2CC2)cc1)NCC1C(NC(C(C)C)=O)CCC1 C1(N(CC)CC)CCN(c2nnnn2C2CC(C(=O)OC)C2)CC1 C(=O)(C1=COc2ccccc2O1)NC(CN(C)CS(=O)(=O)CC1CCOC1)(C)C n1(CCC(=O)NCCC(C)N(C)C(c2ccnc(Cl)c2Cl)=O)cc[nH]c(=O)c1=O c1(CC(=O)N(CC(=O)N(CC(C)(O)C2CC2)C)CC)cnn(C)c1C C1(CC=C)(CNC(=O)C(C)=C2CCCC2)CN(C(=O)CCn2c(C)ccc2C)C1 CS(=O)(=O)c1ccc(S(=O)(=O)NCCc2ccc(C(=O)NCC(N)=O)cc2)cc1 N1(C(c2c(C)nn(C)c2F)=O)CCCC2(NC(c3ccco3)=O)CC2C1 c1(C(=O)NC(C(=O)NCc2cnc(CC)s2)CN(C)C)cc(O)cc(F)c1 Cc1ccsc1CNC(C1CC(CNC(=O)CCN2CCCCC2)C1)=O C(C1c2ccsc2CCN1C(=O)COC)NC(C1(CC#C)CCOC1)=O CCC(C)(C(=O)N1CCOC(CN(C(=O)CCCC2CC2)C)C1)OC C1(CNC(C2C3CN(C)CC32)=O)CC12CCN(C(=O)COC(C)(C)C)CC2 C1(CNC(C2CC(CC)OCC2)=O)CC2CCC1N(C(C1CCCSC1)=O)C2 C12CCC(C)CN1C(=O)CC1(CC1)N(C)C2.C1(CC)CC(OC)C1 c1(NC(c2n(CC)ccn2)=O)ccc(NC(c2cnn(C)c2)=O)cc1C N1(C(C(F)=CC)=O)CCN(C(c2ncn(CC)n2)=O)CC1CC(F)F C12(NC(CCOCC(C)C)=O)CC(C)(C1)OC21CN(C(=O)CCc2ccc[nH]2)C1 C(C(CNC(c1n[nH]c(C)c1C)=O)C(F)(F)F)NC(C1(CCC)CC(=O)C1)=O c1(C(=O)NC2(CC(=O)OC)CCNC2)cc(C(F)(F)F)n(C)n1 C1(NC(c2cc(C)oc2C)=O)CC2CC(NC(=O)COCC3CCCO3)C1C2 c1(OC)c(OC)cccc1CNC(c1cc(CSc2ccccc2)oc1C)=O C1(c2nnnn2C2(COC)COC2)(NCCC=C)CCC2CCN(C2)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(CNC(c2cnn(CCO)c2)=O)C(C)(C)C1 C1(NC(C2C(OC)CC2)=O)CN(C(=O)Cc2cccc(Cl)c2)CC2CCCC12 c1(C(=O)NCC2(OC)CN(C(c3c(OC)ccnc3)=O)C2)ccnc(C#N)c1 c1(C(=O)NC2(CC)CCN(C(COCCC#C)=O)CC2)cc(C)c(N)c(C)c1 c1(CN(C(c2cccnc2)C)C)cn(CCO)c(=O)nc1O N1(C(CCCCCCC)=O)CC2(NC(=O)NCCC(=O)OC)CCCC2(F)C1 C1(C(=O)NC2CCC(C(=O)Nc3cnc(OC)cn3)C2)(CC)CCCCC1 c1(C(N(C(C)C(c2ccccc2)=O)C)=O)cccc2ccoc12 C1(NC(Cc2c(CC)con2)=O)CN(C(c2ncc(N)cc2Cl)=O)C2(CCC2)C1 C1(CNC(=O)COCCc2cscn2)COCCN1C(=O)CCC1CCCOC1 C1(C(=O)OC)(ON2CCC3(CC3)C2)CCC12CCC2 C(C(N=c1ccc(C(F)(F)F)n[nH]1)c1ccco1)OC(C)C CC1(CC(=O)NCCCOCCNC(=O)CC2COCCO2)CCS(=O)(=O)N1 CC(CSc1ccccc1)C(=O)NC1CN(C(C2C(c3ccon3)C2C)=O)C1 N1(C(c2ccnc(C(F)(F)F)c2)C(=O)NCCSC)CCNC(=O)C1(C)C c1(-n2c(C3(c4ccccc4)CCC3)nc(C(CC)O)n2)ccc2nc(C)[nH]c2c1 CC1CCC(C(N2CC(CNC(c3cc(C(F)F)cs3)=O)C2)=O)S1 c1(NC(COCCNC(c2n(CC)c(O)nc2)=O)=O)ccc(C)cc1C CC(C)C(O)C(=O)N1CCN(CC(N2CCC(N(C(=O)CO)C)CC2)=O)CC1 Cc1c(C(N2CC(NC(c3nnc(S)n3C)=O)C3CCCC23)=O)ccc(F)c1F N1(C(CSCC#C)=O)CC(NC(c2ccc(Cl)cc2O)=O)CC(O)C1 C1(O)(C(C)NC(CCNC(=O)OCC)=O)CCN(C(=O)C(O)C(C)(C)C)CC1 c1(CC(=O)NC2CCC(COC)C2)cccc2cn[nH]c12 C1(C(=O)NC2CN(C(=O)C=Cc3cc[nH]n3)CC2C)(OC)CCOCC1 CCC(CSc1ccccc1)N=c1c(C#N)c[nH]c2cc(N3CCOC3=O)ccc12 c1(C=O)cc2ccnc(C)c2[nH]1.n1(CCOC)ccc2ccc(-c3nn[nH]n3)cc12 C1(CC(=O)NCC(C)N(C)C)CN(C(=O)CC2CC(OC(F)F)C2)C(C)(C)C1 C1(C(=O)NCCOCC(=O)NC)N(C(=O)C(C)c2cc[nH]n2)CCCC1(C)C N1(C(Cc2nc(C)[nH]n2)=O)CCCC2(CCCN2C(C2CCCC2(F)F)=O)C1 CN1CCN(C)C(C(=O)NCC(N2CC(F)(COc3ccc(CO)cc3)C2)=O)C1 CCC(C)CC(=O)NCCC(CNC(=O)C(C)(C)c1csc(C)c1)OC c1(NC(c2ccc(C(F)(F)F)[nH]2)=O)cnc(NCC2CC2C(F)(F)F)c(F)c1 N1(C(CC=CC)=O)CCC(CCC(=O)OCC2CCCCN2CC)C(C)C1.OCC C(=O)(C1CCCn2cnnc21)NCC1C(NC(=O)C2=COCCO2)CC1 CC1(C)CC(C#N)(C(=O)NC2CN(C3CC(CNC(=O)C4CC4)C3)C(C)(C)C2)C1 n1(CCCC)nc(C)c(-c2noc(CNC(=O)NC3CC3OC(C)(C)C)n2)c1C c1(C2CCN(C(C3CCOC3)CNC(C)=O)C2)ccc(OC(F)(F)F)cc1 C(=O)(C1CCc2c[nH]nc21)N(C(C)Cc1ccc(F)cc1F)CC C1(NC(CCN(CCC)C)=O)CN(C(C2CCSC2)=O)CC1OC C(=O)(CCS(=O)(=O)NCC)NCC1(F)CC(NC(C(CC)OC2CCCC2)=O)C1 N1(C(CNC(C)=O)=O)CCCCCC1CNC(=O)CN1CCC(C)CC1 N1(C(CCn2cc(CCN(C)C)nn2)=O)CC2(CCOCC2)C1c1cnn(C)c1 C1(CC(=O)NC)CN(C(=O)CCF)CCN1C(c1cc(OC2CC2)ccc1C)=O Cn1ccc(=NC(=O)C2(CCNC(c3ccc(CO)cn3)=O)CC2)[nH]1 S(=O)(=O)(CCC(=O)N1CCC(c2nc(-c3ccc(Br)c(C)c3)no2)CC1)NC C(CCC(=O)NCC1CC(NC(=O)CCc2nnc(C)o2)C1)OCC c1(C(N2CCC(NC(c3c(C)n[nH]c3C)=O)CC2C)=O)oc2ccccc2c1Cl c1(COC)ccc(C(N2CCC(OCCCNC(=O)CC#N)CC2)=O)cc1 C1(CC#C)(C(=O)NCc2cccnc2)CCN(C(c2n[nH]cc2Cl)=O)C1 C(=O)(C(O)CC(F)(F)F)N1CCCC(F)(CNC(c2cncnc2)=O)C1 N1(C(c2nnc(C)s2)=O)CC2CC(NC(=O)Cc3coc4ccccc34)C(C2)C1 N1(C(c2cc(OC)n[nH]2)=O)CCC2(CCC2CNC(C2(SC)CCC2)=O)CC1 c1(OC)ncc(F)c(N2CCC(C(=O)NC3COCCC3(F)F)C2)n1 C12(C(N3CC(C)C(CCNC(c4ccc(C#N)s4)=O)C3)=O)CC(C)(CCO1)C2 c1(C2N(C(Cn3nc(C)c(I)c3)=O)CCCC2)cccc2c1CCCC2 c1(CN2CCC(F)(C(N3CC(C(N)=O)NCC3)=O)C2)ccc2c(c1)OC(F)(F)O2 c1(OCC2C(OCC)CC2)cc(Br)cc(C(F)(F)F)c1O C1(NC(CC2COCC(C)O2)=O)CCS(=O)(=O)C12CN(C(c1c[nH]c(=N)s1)=O)C2 C(=O)(CCCCCC#N)OC(C(C)C)Cc1ccc(F)cc1F C12(C(=O)OCC)CN(Cc3cc([N+](=O)[O-])sn3)CC1CCO2 N(C(=NCCOc1cccc(Cl)c1)NCCCOC1CCCC1)C(C=C)C C(=O)(CC(C)P(C)(C)=O)N1C(C)CC(NC(c2c(CC)n(CC)nc2)=O)C1 N#Cc1ccc(F)c(C(N2CCN(Cc3c(Br)ccnc3Br)CC2CO)=O)c1 c1(CC)cc(C(=O)OC)cc(C(=O)NC2CCC(c3cccc(F)c3)C2)c1 C(C)(C)(CC(F)C(=O)N1CCC2(C1)CN(C)C2)NC(c1ccc(C)nc1)=O C(C(O)C(=O)NCCn1ccc(C(=O)N(C2COCC2O)C)c1)SC c1(C2C(C(=O)NCCCCNC(CC=CC)=O)C2)c(F)cccc1Br CC(CCCC(=O)NCC(=O)N(C)O)NC(=O)COC1(C)CCCC1 CCCCCCC(C)(CC)C(=O)NCCCN(C(=O)COC1CCOC1)C c1(OC)cc(C(=O)NC2CC2NC(=O)CCCNC(C)=O)n(C)n1 C1(O)(CNC(C(C=CC)O)=O)CCCN(C(=O)C=Cc2cnn(C)c2C)C1 C1(C(=O)NCC(C)CN(C(=O)COCc2nc(C3CC3)no2)C)COC(=O)O1 Cc1ccc(C(=O)NC(C)(CNC(=O)CC2COCCOC2)CC(C)C)c(F)c1 Cc1cc(C(=O)N(CCCN(C)C(C2CC3CCC2C3)=O)C)ncc1CO CCC(C(=O)N1CC(C(=O)N(CCC(C)C)CC)(CC)C1)C(C)(C)CC CC1CC(C(=O)NCCCCCCN(C)C)CCN1C(C1COCC1(C)C)=O C#Cc1cccc(CC(=O)N(CCC(C(C)C)NC(=O)CC2CCC2)C)c1 N1(C(C2C(=C)C2)=O)CC(C)(C)CC1CC(=O)NCc1nc[nH]n1 CC1CCc2[nH]c(=NC3CC(N(C)C)C3)[nH]c(=NC3CN(CCF)C3)c2C1 c1(C(N2C(C(NOCCOCCOC)=O)C=CC2)=O)cnccc1OC C(=O)(C(F)C(C)C(F)(F)F)NCC(C)(C)NC(C1=C(C)OCC1)=O Cc1cc2c[nH]nc2cc1C(N1CC(CCNC(c2cc[nH]n2)=O)C(C)C1)=O c1(C(N2C(C(N(CCOCCO)CC)=O)CC2)=O)cnc(C)cc1C C(=O)(C(F)(F)C(F)F)NC1C(NC(=O)CCc2cnco2)CC1 CC(CO)C(=O)NCCCCCN(C(=O)C(C1CCCCC1)O)C C(=O)(CCCC(=O)N1CC(OCCNC(c2c(COC)noc2C)=O)C1)NCC N1(C(C2CCN(C(C)C)C2)=O)CCC(C2CCN(C(=O)Cc3ccon3)CC2)C1 N1(c2c(C(CCC(C)(F)F)=O)cccc2)CCC2(CC1)CC(S(N)(=O)=O)C2 C=CC(CC)CC(=O)NC(CC(F)F)C(=O)N(C1CC(F)(F)C1)C C(=O)(C(CC(=O)N1CC2CCCCC2(c2nnc(C)o2)C1)C(C)=O)OCC CC1(C)CCN(C(c2ccc(Cl)s2)=O)CC1NC(c1cn(CCCF)nn1)=O C(c1ccc(C(N)=O)o1)=CC(=O)N(C(C)=O)CC.C12CCCN1C(=O)C(C)S2 c1(OC)ccc(C(N2CC(O)CC2CNC(=O)CC2(CO)CCC2)=O)c(F)c1 C(=O)(CC(CC)OC)NCCC(=C)CNC(=O)C(C1CCC1)OC C(=O)(C1CCc2c(Cl)cccc21)N1CCCC(CCNC(C2CC(=C)C2)=O)C1 C1(CNC(C2N(C(c3cc(COC)oc3C)=O)CCC2)=O)CCCOC1(C)C C1(C(=O)NCCC(C(C)C)NC(C2CCC(C)CC2)=O)CCCC(C)(C)CC1 C1(C(C(=O)NCCCN(C(=O)C=C2CCC2)CC)C)NC(=O)NC1=O C1(CC(=O)NC2(CC=C)CCN(C(c3cnccc3Cl)=O)C2)CC(=O)NC(=O)C1 C1(NC(CSc2ccc(C)cc2)=O)CC2CC1N(C(=O)Cc1cnccn1)C2 N1(C(CSCCOC)=O)CC2(C=C(C(=O)Nc3cccc(SC)c3)CO2)C1 Cc1onc(CO)c1C(=O)NC(C)CCN(C)C(c1csc(C)c1N)=O CC(C)CC(C)(O)CNC(=O)CN(C(C1CC(OC(C)(C)C)C1)=O)C1CC1 N1(C(c2c(CC)cccc2)=O)CC2(CCN(C(=O)CC(C)C(F)(F)F)CC2)C1 c1(C(N2CC=CC(NC(C(C(=C)Cl)(C)C)=O)C2)=O)ccc2c(c1)C(=O)CCO2 CC1Cc2[nH]c(=NC(C)C3CN(C(=O)OC(C)(C)C)CCC3O)nc(O)c2C1 C1(NC(CCC(CC)C)=O)CCCCN(C(c2sccc2S(C)(=O)=O)=O)CC1 C(=O)(CCCN(C)C)N(CC=CC(=O)N(CC)CC1CCOC1)C C(=O)(C1CCCc2ncnn21)N1C(CNC(C2CC(OC)C2)=O)CC1 c1(C(=O)NC(CNC(CCC(=O)NCCC)=O)C(C)(C)C)cc(N)ccc1C C1(C(=O)NCCc2ccnc(C)n2)CCOCCN1C(C1COCCO1)=O N1(C(C(=O)NC)C)CCC2(CC1)CN(C(=O)CN1CCNC1=O)CC(C)O2 c1(OC)nc(Br)ccc1NC(C1CC(C)CN1Cc1csc(Br)n1)=O C(=O)(C1Cc2ccc(F)cc21)N1C2C(NC(=O)C(F)=CC3CC3)CC(C2)C1 CC1CC(CC(N2CCOC(CN=[N+]=[N-])C2)=O)CN1C(=O)Cc1cc[nH]c1 C1(CC(=O)N(C2CC(CC)C2)C)CCCN(CC(O)COCc2ccco2)C1 c1(C(=O)NC2CC(N(C(CCC(=O)OC)=O)C)C2)cc(Cl)ccc1F C1(CCNC(C2CC(C(N)=O)C2)=O)CN(C(=O)CNc2ccco2)CCO1 C1(CC(=O)NCC(c2nn[nH]n2)C)CCN(C(=O)Cc2cncc(O)c2)C1(C)C c1(NCC2(SC)CCC2)ccc(S(=O)(=O)N2CC(N3CCOCC3)C2)cc1Cl c1(CC)onc(C)c1CN1CCCC1CCNC(c1cc(CSC)c(C)o1)=O c1(SCC(=O)NCCCN(C(=O)CC(C)C(F)F)CC)ccc2c(c1)OCO2 CCC(CC(=O)N1CCN(C(=O)CCC(C)(C)C#N)CC(C)(C)C1)C(C)(C)C C(=O)(C(C)(O)C(F)(F)F)N1CC(OC)C(N)C1.C1(NC(=O)C2CC2)CCC1 c1(C(N2CCC(O)(CCNC(CSCC#C)=O)CC2)=O)ccc2c(c1)C(C)CN2 N1(C(C2CC(=C)C2)=O)CC2(CCCC(CNC(=O)COc3cccc(F)n3)O2)C1 c1(C(N2C(CNC(CN(C)C(N)=O)=O)CC2)=O)cnc(N)cn1 Cc1ccc(CCC(=O)N(C2(CO)CC2)Cc2cn(Cc3cccs3)nn2)cn1 c1(Cn2cc(NCC3(C(=O)OC)CC(=O)C3)nn2)c[nH]c2cccc(C)c12 C(=O)(C1=NOC2COCC12)NC(CC)CNC(c1cnc(C(F)(F)F)c(F)c1)=O CN1CCN(C(=O)CC2(C3CCCO3)CC2)CC1C(=O)NCCF n1(CC(=O)Nc2cccc(C(CC(=O)OC)OC)c2)cc([N+](=O)[O-])ccc1=O c1(C(=O)OC)cnc(N2CCCC2C(C)(C)NC(=O)C(C)O)cc1C c1(-c2noc(C)c2C(=O)NCC2CC(NC(=O)C(F)F)C2)cc(F)cc(F)c1 c1(C(=O)NCC2CCN(C(C(CC=C)(C)N(C)C)=O)C2)cnc2c(c1)CCOC2 c1(C(=O)NC(COCC)C(=O)NC(CO)C2CCC2)cccc(F)c1 Cc1cccc(NC(C2CC3(C2)N=N3)=O)c1[N+](=O)[O-] C=CCC(C)(CC)C(=O)NCC(CCO)NC(=O)Cc1cnccc1Cl N1(C(c2cnc(C)[nH]2)C(=O)NCCCCCC)CCOC(C2(C)CC2)C1 C1(NC(=O)CC=C(Cl)Cl)CC2CC(NC(=O)C(O)CN3CCCC3)C2C1 c1(C(=O)NC2CCN(C(C3C(C)(C)C3(C)C)=O)CC2O)cccc2nc(S)oc12 Cc1sccc1CC(=O)N(C)CC1CCCN1C(=O)CC1CC1CC1CC1 c1(CC)ccc(NC(C2CCC(C(N3CC(OCCN(C)C)C3)=O)C2)=O)nc1 N1(C(Cc2c(C)nn(C)c2)=O)CCC(C(=O)NCC(C)F)C1(C)C c1(OC)ccc(C(N2CCC(c3cnccn3)CC2)C(=O)NCC(F)F)c(C)c1 N1(C(CC(C)(C)C)=O)CCC2(NC(=O)CN=S(C)(C)=O)CC2C1 CCC(C)CC(C(=O)NCCC1CCOCC1)NC(c1cc(O)cc(F)c1)=O CC(CC(F)(F)F)C(=O)NC1CCCC1CN(C)C(C12CCCC1CCC2)=O C1(NC(c2cnn(CCC)c2C)=O)CCCN(C(=O)NC(C)C)CC1F CCC(C(=O)NCC1(COC)CCN(C(c2ncccc2NC)=O)C1)C(F)(F)F N1(C(C(C)C(C)(C)C)=O)CC2CCC(CNC(=O)C(c3ccccc3)F)C2C1 N1(C(=O)Cc2ccco2)CC2(CC(C(N3CCC(C(F)F)C3)=O)CO2)C1 N1(C(CCCOC)=O)CCCC(NC(c2cnn(CCO)c2C)=O)C(F)C1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NC(CC(C)NC(c1nc(C(C)C)oc1)=O)C N#Cc1cc(S(=O)(=O)N2CCC(CC(=O)Nc3cccnc3Br)C2)ccc1F c1(OC(C)(C)C)ccccc1C=CC(N1CC(CCF)C1)=O C(CCC(O)C(=O)NC1CCC(C(N)=O)C1)NC(c1cc(C)sn1)=O C(=O)(C1=CCCN(C(C2(C)CC(F)C2)=O)C1)N(CC#C)CCOC N1(C(c2cn(CCC)nc2)=O)CCC(F)C(NC(=O)CN2CCC(CO)CC2)C1 C1(CCC)C(C)CCCN1C(C1(CNC(=O)CC2CC(C)=NO2)CC=CC1)=O C1(C(N(CCn2cncn2)CC)=O)CC(NCC)C(O)C1.c1(C(=O)N)ccsc1 Cc1nn(C(C)C)c(C)c1C(N1CC(NC(c2cc(C#N)no2)=O)C(C)(C)C1)=O C1(CC)(NC(c2ccc(Br)nc2)=O)CCN(C(=O)C(C)Cc2ccccn2)CC1 c1(NC(C2CC(C(F)F)(OC)C2)=O)ccc(NC(=O)CN(C)C(C)C)c(C)c1 c1(C(N2CCCC(c3cn(CC(=C)CC)nn3)C2)=O)cnc(O)n(C)c1=O C(=O)(CCCCCCS(N)(=O)=O)NCC(C)CNC(=O)COC1CCN(C)CC1 C1(C(=O)NCC(C(=O)N(CC(O)CF)C)O)CC(=O)NC(=O)C1 C1(CN(C)Nc2cc(Oc3c(OC)cccc3)ncn2)CN(C)CCC1(F)F C1(CC)CCCC1C(=O)NCC(C)(C)CNC(=O)CSCC#N c1(C(=O)NC(C)CC(C)NC(=O)C(C)Cc2cnn(C)c2)cnc2ccccn12 c1(C(N2CC3C(CNC(=O)Cc4sc(O)nc4O)(C3)C2)=O)cc2n(n1)CC(F)C2 C12(CNC(c3n(CCC)ccc3)=O)CCCN(C(=O)Cn3ccnc3C)C1C2 Cc1cc2c(cc1C(=O)N(C)CC1(O)CN(C(C3CC34CCOC4)=O)C1)OCO2 c1(C(=O)NC2C3CN(C(C4(F)C(C)OCC4)=O)C2C3)cc2n(n1)CCOC2 C(=O)(C(F)(F)CN1CCOCC1)OC(c1cccnc1)C(=O)OC c1(C(=O)NCC2(CN(C(C3C(C#C)C3)=O)C)CC2)cccc(N)c1Br c1(C(=O)NCC2CCN2C(c2cnc(C3CC3)s2)=O)nccc2ccccc12 c1(N2CC(C(C(=O)CC(C)CN(C)C)C)C2)ncc(C(F)F)cn1.C1(=O)C(C)(C)N1 S(=O)(=O)(c1c[nH]c(C(=O)NCC2CN(c3ccccc3)C(=O)O2)c1)N(C)C C1(CN(C)C)CN(C(C2(C(=O)NCc3c(N(C)C)n(C)nc3)CC2)=O)CC12CC2 N#Cc1ccc(Br)c(C(=O)NC2CCC(NC(=O)Nc3ccc(F)nc3)C2)c1 Cc1cc2nc(NCC3C(C)CCCN3C(=O)CN(C)CCO)cc(=O)n2o1 c1(CC(C)(C)C)ccccc1C(N1CCOC(CNC(C23CSCC2C3)=O)C1)=O N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(O)CNC(=O)CCF c1(OC(C)C)ccc(C(=O)N(C)CCCOC(C)C(=O)Nc2ccccc2)cc1N CC(C)C(F)C(=O)N1CC(CNC(c2cnncc2O)=O)C(O)C1 c1(OC)cccc(N2CCC(N(C)C(c3sccc3F)=O)C2)c1CO C(=O)(C1=NOC(C)(C)C1)NC1CN(C(CCc2nc(C)c(C)[nH]2)=O)CC1(C)C C1(C(=O)NC(CC2CCN(C(c3nc(C)oc3C)=O)CC2)C)CCCCS1(=O)=O c1(C(=O)NC(C)CCCNC(c2cc(CO)[nH]n2)=O)c2ccccc2nn1C C(CCC(=O)N(C1CC(NC(=O)C(C2CC2)N(C)C)C1)C)=CC(C)C CON(C)C(=O)C(CC1CC1)CC1CC1.C(=O)(C(F)(F)C(C)(C)O)N C(=O)(C(O)P(C)(C)=O)N1CCCC(CCNC(c2cc(COC)on2)=O)C1 N1(C(CC=CCCCCC)=O)CCC(C(=O)NCCOCCCO)(CF)C1 C1(N(C(CC(=C)Br)=O)C)CCCCC1N(C)C(c1csc(CC)n1)=O C1(NC(CSCC)=O)CC2CN(C(=O)CC3CCC(C)(C)CC3)CCN2C1=O c1(C(C(=O)N(CCN(CC)CC)C)NC(=O)CCn2cnnn2)cn(C)nn1 N#Cc1ccc(C(c2nnnn2CC2CCCO2)Nc2cccnc2C(N)=O)o1 c1(C(C(=O)NCCCCCn2cc(CCCOC)nn2)C)cccc(OC)c1 Cc1cc(Cl)ncc1CC(N1CC(NC(=O)C(C)(C)OC(C)C)CCC1C)=O C(C(C)CC(C)C)NC(c1n(CCCSC)nnn1)c1cscn1 C(=O)(CCCCCCNC(=O)CC1CCCOC1)N1CCC(C#CC)C1 N1(C(C=C(C)C(C)C)=O)CCC(NC(=O)Cc2cn(C3CC3)cn2)C1C c1(C(=O)NC(C)C(C2CCCCC2)NC(=O)C=CBr)ccnc2[nH]nnc12 C(=O)(C1=C(F)CN(C(=O)CC(C)SCC)CC1)NC1(CC=C)CCCC1 Cc1nccc(=NC2CCC3CN(C(c4cn(C)nc4C(C)C)=O)CC23)[nH]1 C1(CNC(C(C)(C)OC)=O)CN(C(C2CCC(O)C2)=O)CCC12CCC2 O=[N+]([O-])c1cccc(NCCOS(=O)C2COC2)c1 C(=O)(C(CC(C)(C)C)N1CCCC(C(F)F)C1)NC(CC)(C)C C1(C(N(CC(C)(C)C)CCC)=O)CC(F)CN1C(C1CCCC1OC)=O CCC(C)(C)C(C)NC(c1coc(C(C)NC(=O)C=CCN2CCC2)n1)=O c1(C(N2CCC(C(C)NC(c3c(C)cn(C)c3)=O)C2)=O)cc(Cl)ccc1C(F)F C1(NC(C2CCCC(C)(C)CC2)=O)CC(N=c2ccnc(N3CCOCC3)[nH]2)C1 C(=O)(CC(C)(C)C(F)F)N1CC(O)(CCNC(C2(C)CNC(=O)C2)=O)C1 N1(C(C(CSC)(C)NC(c2ccc3[nH]ccc3c2)=O)=O)CC2C3CCC(C3)C2C1 N(C1c2ccccc2CC1NC(C1CCS1(=O)=O)=O)C(CN(C)C)=O n1(CC)cnc2c(NCC3CS(=O)(=O)CCO3)[nH]c(=NCCC(C)N(C)C)nc12 CC1(C)CC=C(C(=O)N2CCC3(CC3NC(C3CCOC3)=O)C2)CC1 CCCN=C(NCCN1CCCOCC1)NCc1conc1CC Cc1noc(CCN2CCC(N3CC=CC3)C2)n1 Cc1ccncc1C1(NC(c2csc(-c3ccncc3)n2)=O)CC1 C1(CC)CN(C(=O)CCF)CCC1NC(=O)COc1cnn(CC2CCCC2)c1 N1(C(C(CC(F)F)N(C(COC(C)=O)=O)C)=O)CCc2nncn2CC1 N1(c2ncc(C)cn2)CCC(NC(=O)C(F)(F)C2CC2)C(CO)CC1 c1(CNS(=O)(=O)C(F)F)cccnc1-c1ccc(C2(NC3CC3(Br)Br)COC2)cc1 C1(NC2CC(CC(=O)OC)C2)CCc2nn(C)c(C(=O)O)c2C1 c1(C(N2C(CNC(CC3CC(=C)C3)=O)CC2)=O)cc(S(N)(=O)=O)oc1C C1(O)(C(C(=O)NC)(F)F)CCN(C(=O)C(=O)Nc2cnn(C(C)C)c2)C1 C1(CCOC)(NC(C(C=C)(C)O)=O)CCN(C(=O)COc2ccsn2)CC1 C1(C2CCCN(C(C3CCCCC3C3CC3)=O)C2)(NC(CN(C)C)=O)CC1 C1(C(=O)NCCN(C)C(c2ccc(F)cc2O)=O)COC2(CCC2)C1 c1(CC)cccc(C(N2CC(O)(CNC(C3CC(C4CC4)=NO3)=O)C2)=O)c1O N1(C(c2c(CCC)n[nH]c2)=O)CC(C)C(C)(C(N2CCC(C)=C(C)C2)=O)C1 N1(C(C(C2CCOC2)OC)=O)CCC=C(CNC(c2ccc(C)nc2C)=O)C1 C1(C(=O)NC2CN(C(CC(CCSC)O)=O)C2)Cc2ccccc2S1 C(C)(C)(C(=O)NC1CC1CNC(=O)CCCOCCOc1ccccc1)OC N1(C(c2cn(CC)nc2)=O)Cc2n[nH]cc2C1C(=O)NCC1CC(SC)C1 C12(NC(C3N(C(C)=O)CCC3)=O)COC(C1)C(NC(=O)CSCC(C)C)C2 Cc1coc(C)c1C(N1CCC(CN(C(=O)C(c2ccccc2)C2CC2)C)C1)=O N1(C(C2CC(C)(F)C2)=O)CC2CCC2(CC(=O)NC2CC23CCCC3)C1 C(=O)(C1=Cc2ccccc2OC1C(F)F)NCc1cn(CCCC(=O)O)nn1 [N-]=[N+]=Nc1cncc(C(=O)Nc2ccccc2-n2cc(-c3cscn3)nn2)c1 N1(C(C2N(CC)CC2)=O)CC(CNC(=O)C(c2ccc(F)cn2)(F)F)CC1(C)C Cc1ccc(N2CCC(N3CCC(NC(=O)CC4CCSCC4)C3C)C2=O)cc1 CC(CNC(=O)N(Cc1cccs1)CC1CC1)CC(F)F Cn1nc(-c2ccncc2)cc1C(N1CC(n2cc(C3CC3CO)nn2)C1)=O N1(C(CSc2nc(C)sc2)=O)C2CCC1CC(CNC(C13CC(CO1)C3)=O)C2 c1(COC)csc(CN2CCCC2C(c2ccccc2)C(=O)NCC)n1 n1(CCC(=O)OC)cc(C#CCNC(=O)C(c2ccc(SC)cc2)C)nn1 N1(C(C2C(C)C2)=O)CCc2ccccc2C(NC(C2CCC(OCC)CC2)=O)C1 C1(C)CCCN(CC(=O)N(CC(C)C)C)C1.Cc1cc(NNC2CC2)no1 C(=O)(CCN=c1[nH]c(C)cc(=NC(C)c2n[nH]c3ccccc23)[nH]1)NC C1(NC(C(CC)C)=O)C2CC(O)C1N(C(=O)C1=CSCCO1)C2 CCCC(C)C(=O)N1CCC(Cc2cc[nH]c2NC(C2COC2)=O)CC1 N1(C(C(c2cc(C)sc2)(F)F)=O)CCN(C(C2(C)CCCC2)=O)C2CCCCC12 CC(C)(C(=O)N1CCC(c2ncco2)C1)C1=CCN(C(C2(C)CC2(C)C)=O)C1 C1(C)(C(=O)NCC(CC)NC(c2cc(C(C)C)no2)=O)CCCOC1 C1(CC(C(C(=O)OC)C)=O)CCN(C(=O)OC)CC1 C(CO)(C(=O)NC(C(N)=O)C1CC1)NC(CN(C)C1CC1)=O c1(C(C(=O)NC2C3CCN(C(c4cc(C5CC5)no4)=O)C23)O)ccc(Cl)cc1Cl C1(CC(N2CC(OCCNC(CCc3c(C)ncs3)=O)C2)=O)CCCCN1C C(=O)(C(C(=O)N=c1ccn(CC(=O)OC)[nH]1)C(C)C)OCC c1(C(N2CC(CC)N(C(=O)CCNC3CC3)CC2)=O)cc(OC)c(O)c(N)c1 c1(OC)c(C(N2CCC(CNC(C3COC(=O)C3)=O)CC2)=O)occc1=O C(=O)(C1=CC2CCCC12)NC1(CNC(c2ncc(C)cc2C)=O)CCC1 c1(C(=O)NC2CC(C(=O)O)C2)cccc2c1CCS2(=O)=O c1(NC2C(C)CN(C(=O)Cn3cnnn3)CC2C)nc2cccc(F)c2s1 C1(CNC(C2CC3CCCCN3C2)=O)CCCC2(CN(CCCC3CCC3)C2)O1 C(=O)(C(O)C(F)(F)F)N(CCCNC(c1c(C)nc(C(C)C)[nH]1)=O)CCO N1(C(c2cn(C(C)C)nc2)=O)CC(C)CN(C(C2CCOC2)=O)CC1C c1(CN2C(C3(O)CN(C(C(C)(C4CC4)NC(C)=O)=O)C3)CCC2)cc(O)nc(O)c1 N1(C(C(C(CC)C)O)=O)CCC2(CC1)CCN(C(=O)CCOC(C)C)C2 C1(NC(=O)CNc2nccs2)COCCC1CNC(=O)CN1CC(=O)NC1=O N1(C(C2CCC(F)(F)C2)=O)CCOC2(C1)CN(C(=O)C(c1ccccn1)O)C2 c1(OC)ccc(C(=O)NCC2CCCC2NC(=O)C(C)C(F)(F)F)c(O)c1 C1(C(=O)NC2C(NC(c3cn(CCO)nn3)=O)COCC2)CC2CC1C1CC21 Cc1cc(-c2c[nH]c(=NCc3c[nH]nc3C(F)(F)F)s2)ccc1CN(C)C CC1=CCC(C(N2CCCC2(C)CNC(=O)CC2CC(=O)NC2=O)=O)CC1 N1(C(C(C)=O)=O)CC(NC(c2ccc(C)n2C)=O)CC2(CCC2)C1 c1(C(=O)NCC(C)NC(=O)CN2CCOC2=O)cc(S(N)(=O)=O)oc1Cl c1(C(=O)NCC2N(C(COCC(C)C)=O)CCC2)ccc(OC2CCC2)cc1 N1(C(C(C)OCC)=O)CCC(C)(CNC(=O)CC2CCCN(C)C2)CC1 CCC(O)CCc1cn(CC(F)CCNC(=O)Cc2cccn2C)nn1 c1(CC)c(C)nn2c(C)cc(C(=O)NC(C(F)F)C3CCCOC3)nc12 c1(C(N2CCC(C(C)NC(C3CC4CC3C4)=O)CC2)=O)nn(C)c2c1CCC2 CCCC(O)CC(=O)N1CCC(C)(NC(C2CCCCC2n2cccn2)=O)C1 c1(C(=O)NC(CC(=O)NCc2n(CCC)cnc2)C2CC2)cn(C)c(C)n1 CCCCC(CC(=O)N(C(C)CO)C1CC1)NC(=O)Cn1cnnn1 NS(=O)(=O)c1sc(N2CCCC(NC(=O)NCCC3CC4CCC3O4)C2)nc1Cl C1(C(=O)NCCC2CCC(NC(CNS(N(C)C)(=O)=O)=O)C2)CN(S(N)(=O)=O)C1 C1(C(N(C(C)C)CCN(C)C(C2CC(=O)C2(C)C)=O)=O)CCCNC(=O)C1 c1(OC)cc(C(=O)NC(C)C(C)NC(c2ccnc(CO)c2)=O)cc2c1OCC2 C1(CC(C)NC(=O)C=Cc2cscn2)CCN(C(c2c[nH]ccc2=N)=O)CC1 C1(CNC(COCC(C)C)=O)CC(O)C(O)CC1C(N1CCC(F)CC1)=O C1(NC(c2cncc(OC)n2)=O)CN(C(=O)C(c2ccccn2)C)CC1C1CC1 C(C(C)C(=O)N1CCCC1CC(=O)NCC(N1CCOCC1)=O)SC CC1OC2(C)CC1(C(N1CCC(OC3CN(C(=O)C4=CCOCC4)C3)CC1)=O)C2 N1(C(C2C3C(NC(C4CC4Cl)=O)C4C(C3)C42)=O)CCOC2CCC12 Cc1cccc(-n2cc(C3(C)CCCO3)nn2)c1 N1(C(C2N(C(CN3C(=O)CCCC3)=O)CCC=C2)=O)CCC2CC1C(=O)O2 C(CC(C(C)(C)C)NC(C1(C(=O)OC(C)(C)C)CC1)=O)N(C)C(C1CCCC1)=O C1(CCNC(=O)Cn2cc(Br)cn2)COCCN1C(C12CCC1C2)=O c1(C(c2nnnn2CC2CC2)NC(C(C)C)C2CCC2)csc(C2CCCO2)n1 c1(CC)ccc(C(C)C(=O)N(C)CC2CCCN2C(C2(C(C)C)CC2)=O)cc1 N1(C(CCOCC)=O)CC(NC(=O)CC(c2ccccc2F)NC(C)=O)C(C)C1 Cc1cc(C(=O)NC23COC(CNC(C4CCC(C)C4)=O)(C2)C3)sc1C C1(CS(=O)(=O)NC(c2cccc(Cl)c2)C(=O)OC)CC2(CCC2)CO1 c1(C(=O)NC2(C3N(C(C(CC)SC)=O)CCC3)CC2)cccc(Br)c1F Cc1cc(C(N2CCC(C)C(NC(C3CC3(F)F)=O)C2)=O)cc(C)c1O c1(OC)ccc(C)cc1C(=O)N(C1CCCN(C(=O)Cc2ccc(C)nc2)C1)C C1(NC(C2CCC(=O)O2)=O)COCCN(C(=O)Cc2cscn2)C1 c1(OC)ccc(CCC(=O)NC(C2CCN(C(C)=O)C2)C)cc1 C1(N(C(C=CC=CCC)=O)CCO)CCN(C(=O)CCc2ccc(C)s2)CC1 C(=O)(N=[SH](C)(CCN)C(C)(C)C)c1ccc(CC)cc1 N1(C(c2c(C)nn(CCO)c2)=O)CC(CNC(=O)CC2C=CCCC2)CC(C)C1 c1(CCOC)nc(C)c(CN2CCCC(CNC(=O)Cc3ccsc3)C2)o1 N1(C(C(CC)CC)=O)CCCC(O)(CNC(C2CCOC2Cc2ccccc2)=O)C1 C1(NC(=O)CNC(c2ccoc2)=O)CCCCCN(C(=O)CCCF)C1 c1(OCC)cccc(CC(=O)N(C)CCN(C)C(C2CC=CCO2)=O)n1 C1(CNC(c2cc(C)oc2)=O)C2CCC(C2)N1C(=O)C(C)c1ccsn1 N1(C(C(COC)(C)C)=O)CC2CC(NC(c3c[nH]cc(Cl)c3=O)=O)CC2C1 CC1(C)CCCC(C(=O)NCCCNC(=O)CNS(=O)(=O)c2cccnc2)CC1 C1(CC=C)(C(=O)NC2CCN(C(=O)CCCc3ncc(C)o3)C2)CCCCC1 C1(CSC)(CNC(=NC)NCCCNC(C2CCC2)=O)CCCCC1 N(C(=NCC(C)(C)OC(C)C)NCCC1OCCC1(C)C)C1CC(C)C1 N1(C(C(CCC)OC)=O)CCN(C(=O)C2=CCOC2)CC1C c1(C(=O)NC(CC)CNC(=O)C=CC(c2cnn(C)c2)=O)c(C)noc1C(F)F N1(C(c2cc(C3CCOC3)[nH]n2)=O)CCC2CCN(C(=O)C(F)=CC3CC3)CC2C1 Cc1cn2cc(NC(=O)CCCn3cc(CN4CCC(C(=O)O)C4)nn3)nc2s1 S(=O)(=O)(c1cccnc1NCC(O)C1CCC1)N1C(CSC)COCC1 CCCCC(CNC(c1sccc1NS(C)(=O)=O)=O)NC(=O)C(C)C(C)O C1(CC(=O)NC2C(NC(c3c(C(=O)OC)cco3)=O)COC2)CN2CCC1CC2 C(N(C)N1CCC(N2CCNC2=O)CC1)C1CCC(CCCC)CC1 C1(N(C(c2cnc(C(C)C)[nH]2)=O)C)CCN(C(C2(F)CC=CCC2)=O)CC1 C1(CC)COCC1NC(=O)C(Cn1cccn1)NC(=O)CCn1cnc(=N)[nH]1 N1(C(CC2(OC)CC2)=O)CCC2(CC1)CC(CNC(c1csc(C(C)=O)c1)=O)C2 C(CCC(=O)NC(C)CC(C)NC(c1ccn(CCN(C)C)n1)=O)OCC CC(F)(F)CCCC(=O)N1CC2CCCC1C2CNC(c1cscn1)=O c1(C(C(=O)NC)N(C)Cc2ccc(F)cc2C)c(Cl)nc2sccn12 c1(C(=O)NCC2N(C(C=CC=CCOC)=O)CC3CC32)ccc(N)c(F)c1F C(=O)(C1CCc2ccc(C)cc21)NCC1CCN(C(c2nn(CC)nc2C)=O)C1 N1(C(CCCc2ccc(CCC)cc2)=O)CCCC2COCC12 C1(C(=O)NCC(CNC(c2nnn(C)c2N)=O)(C)C)CCCCS1(=O)=O CN1CCCCC1C(N1CC(C)(OCC(=O)N(C)CC2CCCC2)C1)=O N1(C(CN(C(=O)OC)C)=O)CCCC2CN(C(c3ccn(C(C)C)n3)=O)CCC12 C(C)(CC(=O)NC(C)CC(=O)NCCC1(CO)CCCC1)=C(C)C C(=O)(C#CC1CCOCC1)N1CC(NC(c2oc(C)c(CO)c2)=O)C(CO)C1 C(=O)(C(C(C)CC1CCC1)N1CCC(SC(F)F)CC1)NC(C)C c1(C(C(=O)NCCF)N(C)C2CC2)ccc2c(c1)OC(C)(C)O2 C1(C(=O)NCC2CN(C(CC3C(OC)CC3)=O)C2)CCn2c(Br)cnc2C1 C(=O)(CC(CN(C)C)C(F)(F)F)NCC1N(C(c2c(CC)[nH]cc2)=O)CCC1 C(=O)(C1=CCc2ccccc21)NC1CCCCN(C(C(C)C(F)F)=O)C1 c1(C(=O)NC(C2CCCN(C(=O)Cn3cccn3)C2)(C)C)nnc2ccccn12 N1(C(COC)C)CCN(C(C)=O)CC(O)C1.c12ccc(OC)c(c1)O2 c1(CNC(C2=NNC(=O)CC2)=O)nc(=NC2CN(C(C3CC3(Cl)Cl)=O)C2)cc[nH]1 CC(CN(C)C)CCC(=O)NCC(C)CNC(=O)CCCc1cccc(Cl)c1 C1(NC(CCNC(Cn2ccc(C)n2)=O)=O)CCSC(C)C1 c1(C(=O)NC(C2OCCN(C(C(C)SC(C)C)=O)C2)C)cc(Cl)nnc1O NC1CCC2(C(=O)NCC3CCCNCC3)CCC12 N1(C(C2CC(SC)C2)=O)CCOCC(CC2(C(=O)NCC3CCCCC3)CC2)C1 C(C(C)CC(=O)NCC(C(C)C)NC(c1nn(CC)nc1C)=O)OC Cc1cc(CC(=O)NCC#CCNC(=O)C(C)(C)c2ccc(Cl)s2)n[nH]1 c1(OC)ccc(C(N2CC(CNC(C3COC(C)(C)CO3)=O)C(C)C2)=O)cc1F c1(C(=O)NCC(CNC(C(CC(C)C)F)=O)(C)O)cc(Cl)c2n[nH]cc2c1 c1(C(=O)N=c2[nH]nc(C(F)(F)C(F)(F)F)s2)cc2cc(F)ccc2oc1=O C1(NC(CC(CC)(C)C)=O)CCN(C(c2cccc(C(C)=O)c2)=O)CCC1CO c1(C(=O)NC(C2CN(C(C3(NC)CCCC3)=O)C2)C)cc2sc(C)cc2s1 N1(C(C=CCC)=O)CCCC(C(C)NC(=O)Cn2ncccc2=O)C1 c1(C(C(=O)NCC=C)N(CCF)CCOC)ccc(C(F)(F)F)cc1F Cc1nc(N2CC3CC2(CNC(=O)CC2COC(C)(C)C2)C3)[nH]c(=N)n1 c1(OC)c(C(=O)NCCN(C(=O)CC2COCC(C)(C)O2)C)ccnc1Cl C#CCCC(O)C(=O)NCC(CO)NC(=O)Cn1cc(Br)c(=N)[nH]1 N1(C(=O)NCC(F)CC2CC2)CCC(C(F)(F)CO)C1 c1(NC)ccc(C(=O)NCCCC(C)(C)NC(=O)C(C)CC(C)C)cc1F c1(C(=O)NC2CN(C(CS(CC)=O)=O)CC23CC3)cccc2c1OCC2 C(=O)(CC1OCc2ccccc21)N1CCC(NC(CCC=CCC=C)=O)C(O)C1 N12CCN(CC1C1CCC1)C(=O)C(O)CCC2=O.N=c1ccc(CO)n[nH]1 C1(NC(C)=O)CCN(CCN(S(C)(=O)=O)C)C(C)C1 C(CC1CC1)(C(=O)N(C)Cc1ccns1)NC(CNC(CCC)=O)=O c1(C(N(C)CC2(O)CCCN(C(=O)C(F)(F)C(F)F)C2)=O)cccc2ccnn12 C1(NC(C=C(CCC)CCC)=O)CCN(C(C2CCN2CC)=O)C12CCC2 C(=O)(C(F)(F)CNC(=O)C(CNC(C1(C)CCN(C)C1)=O)N(C)C)OCC N1(C(c2ccc(OC)o2)=O)CCN(C(C2CCC(=O)N(C3CC3)C2)=O)C(C)C1 C1(C(N2CC(C)(NC(CCC=CC(C)C)=O)C2)=O)CC(F)(F)C1(C)C C1(C(=O)NCC#CC2CC2)CCC(O)CN1C(C1CCCC(=O)C1)=O CC(CC(=O)N1CCN(C(C2(C3CCCO3)CC2)=O)CC12CCC2)CC(C)(C)C c1(C(=O)NCCN2CCCC2)ccc(SC(F)(F)F)o1.C12CN(C1)C(=O)CN2 C1(N(C(c2c(CC)nn(C)c2)=O)C)CN(C(=O)CN2CCOCC2=O)CC12CC2 S(=O)(=O)(c1ccccc1)NCC(=O)N(CC(O)CNC(C1(F)CC1)=O)C C1(NC(C=C(C)C)=O)CC(C(F)C(=O)NCC(C)N(C)C2CC2)C1 c1(OCC)ccccc1C(N1CCCC(C2CCCCCO2)C1)C(=O)NC(C)C CC1C(C(=O)N(C)CCN(C(=O)CCc2ccc(C(F)F)cc2)C)CCN1C C1(NC(CC(CC#C)NC(c2cnc(C)o2)=O)=O)CC12CCCCCC2 c1(CNC(COC2(C#C)COC2)=O)cccc(C(=O)NC(CSCC)CO)n1 N1(C(c2nc(C)[nH]n2)=O)CCCC(CCC(=O)NC2(CCN(C)C)CC2)C1 c1(C(C)C)nn(C)cc1C(=O)N(C)CC1C2CN(C(C3CCOC(C)C3)=O)CC12 c1(C(=O)NC(CCC)C(=O)N2CCSC(C)C2)ccc(C)c(C#N)c1 C(=O)(C1=CS(=O)CCC1)NC(C(C)C)CNC(C1CC(n2cnnc2)C1)=O N1(C(C2C=C(C)CS2)=O)CC2(CCN2C)C1.c12cn(nn1)C1CN(C1)C2 CC1C(C(=O)N(CC(C)C#N)C)CCCN1C(=O)C#CC1CCC1 c1(C(=O)NCC(CC)NC(C2C(=C)CC2)=O)cc([N+](=O)[O-])cc(Cl)c1NC Cc1c(C(=O)Nc2ccc(Cl)c(-c3nn[nH]n3)c2)cccc1Br N1(CCNC(=O)NCCc2nccc(OCC)n2)CCc2sccc2C1 N1(C(c2cn(CC(=O)N(C)C)nn2)=O)CCN(C(=O)C(C)(C)C#N)CC1CCO CC1COC(c2ccc(Br)cc2)CN1C(C1(N(C)C(=O)OC(C)(C)C)CC1)=O c1(C(=O)NCCCN(C(CCn2c(C)cc(C)n2)=O)CCO)ccc(C)c(F)c1 C1(NC(C2C(C)(C(F)F)C2)=O)CC(CNC(=O)Cn2cnc(C(N)=O)n2)CC1O CC1CCN(C(=O)CCn2cnnn2)CC1CNC(c1cnc(C2CC2)[nH]1)=O N(C(=NC)N1CC2C(C(F)F)C2C1)CC(c1c(OCC(=C)C)cccc1)C c1(CC)cnc(CC(=O)N(CCCN(C)C)C2CC2)[nH]1.C12CCC(C1)C(=O)N2 N#CCCCC(=O)NCC1CCCC1NC(=O)CCc1cnc(C2CC2)o1 Cn1cnn(CCC(=O)NC2CC2CNC(=O)C(CO)NC(=O)OC(C)(C)C)c1=O C#Cc1ccccc1CN1CC2CC1C2C(=O)Nc1cc(Cl)ccc1C(N)=O C1(CNC(c2sc(C)c(O)n2)=O)CCC(C)CN1C(c1cnn2c1OCC2)=O C1(C(=O)NC(CNC(C(CC)O)=O)C2CC2)CCc2c(nnn2CC)C1 n1(CCC(=O)NCCC2(CNC(C34CC(F)(C3)C4)=O)CC2)ccc2ccccc12 c1(C(=O)NCC2CC3(CO2)CN(C(C2C=CCC2)=O)C3)cccc([N+](=O)[O-])c1Cl C1(CCNC(C(C)OCC=C)=O)CCN(C(c2ccc(OC(F)F)cc2)=O)CC1 CN1CCN(C(=O)CC2CCCN(C(=O)C(C)(C)C3CC3)CC2)CC(O)C1 N1(C(CNC(c2ccccc2)=O)=O)CCCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1 c1(COC)nc(NCCc2csnn2)cc(=NCC2(C3CC3)CC2)[nH]1 Cc1c(F)ccc(C(=O)N(C)CCN(C(C2CN(C)CC(C)O2)=O)C(C)C)c1N N1(C(C2CN(C)C(=O)N2)=O)CCC2(CC1)CCN(C(=O)CC1CCCO1)CC2 C1(CN(C(=O)CN(C)S(=O)(=O)N(C)C)C)CN(C(=O)CCC2CCC2)CC12CC2 c1(NC(C(=O)NCC(CO)NC(C(CC2CC2)OC)=O)=O)cc(C)ccc1Cl c1(OCC(=O)NCCC(CNC(=O)C=Cc2cccnc2)O)ccc(F)c(Cl)c1 N1(C(c2c(C)nn(C)c2Cl)=O)CCC2(CC1)OCCC2NC(C1CC=CC1)=O N1(C(CCC(=C)C)=O)CCC2CCN(c3nc(-c4nccs4)ncc3C)CC2C1 C1(C(=O)NCCCCCCN(C(C(c2cccnc2)C)=O)C)CCOCC1(C)C N1(C(C(CCC)O)=O)CC2(CCCCN(C(c3ncoc3C3CCCO3)=O)C2)C1 c1(C(N(CCCNC(Cc2cn(CC)nc2)=O)CCO)=O)cc(C(F)(F)F)ncn1 c1(C(N2CC(O)(CCNC(c3c(C)cc(C)o3)=O)C2)=O)c(C)ccc(Cl)c1O c1(CNC(C2(NC(C)=O)CCC2)=O)cccn1C1(C(=O)NC(=O)C2CC2)CCCC1.C1(C)CC1 N1(C(C2(CC=C)CC=CC2)=O)CC2ON=C(CNC(c3cnc(CC)s3)=O)C2C1 C1(C(N(C2CCCN(C(COCCOC)=O)C2)CCO)=O)OCCN(C)C1=O Cc1cc(NC2CCCCC2NC(=O)CSC(F)(F)F)ccc1[N+](=O)[O-] C=C(CNCC)C(F)(F)F.c1(C2c3nnnn3CCN2)cc(F)ccn1 c1(C(=O)NCC2(CN(C(C3C(C=C)C3)=O)C)CC2)cnc(O)c(Cl)c1 C1(C(=O)Nc2cn(C(C)C)nc2)(NC(=O)CN2CCOCC2)CCCC1C C(=O)(C1=NOC(C)C1C)NC1CCN(C(COc2cc(C)cc(C)c2)=O)CC1O N1(C(c2cc(CNC(CCc3n(C)cnc3)=O)on2)=O)C2CCC1CC(CO)C2 Cc1nccc(NC(=O)CN(C2CCCNC2C)C)n1 C1(NC(CCC2CCCN(C(C3C(OC(C)=O)C3)=O)C2)=O)CCNC(=O)CC1 Nc1ccc(Br)cc1C(=O)NC1(CNC(c2cnn(CCCF)c2)=O)CC1 c1(C(N2CC3C(NC(c4ccc(C(C)(C)C)[nH]4)=O)C3C2)=O)cc(F)cnc1O C1(C(=O)NC23CC(NC(c4c(C)nccc4)=O)C(OC2)C3)CNC(=O)C(C)(C)C1 C(CCCCC(=O)NCC1(F)CN(C(=O)C(F)C2CCC2)C1)OCC c1(C(N2C(C)CC(NC(C3(COCC)CC3)=O)C2)=O)cc(C)c(F)cn1 CCC(C)(C)CC(=O)NC1CCC(CCNC(c2ccc(C)c(N)c2)=O)C1 c1(C(=O)OC)cc2c(s1)CCC2NC(=O)CN1CCOC(c2cc(Cl)cc(Cl)c2)C1 Cc1ccc(=O)n(CC(=O)NCC(C)(C)NC(c2conc2C2CCCO2)=O)c1 N1(C(CNC(=O)NC)=O)CCC(NC(c2cncc(C)c2Cl)=O)CC1C1CC1 C#Cc1cccc(C(=O)NC2CC2NC(=O)C(O)CC2CCCC2)c1Cl CC1CCCCCC1NC(C)Cc1cccc(F)c1 CC1CC(=O)NCCN1C(c1cc(Br)co1)C(=O)NCc1ccc(F)cc1 C(CCCCCCCO)=CCNC(C1N(C(CC(CC)C)=O)CC(F)C1)=O c1(C(=O)NC2C(CC)CN(C(=O)CSC3CC3)CC2)cc(S(C)(=O)=O)ccc1F C1(C(=O)NC(c2ccccc2)C)C2Cc3ccccc3C12.C1(=O)C=CCO1 N1(CCC)CCC(C(=O)NCCN(c2ncc(Cl)cn2)C(C2CCCC2)=O)CC1 c1(NC(C(Cc2ccoc2)NC(=O)CCn2cnnn2)=O)cccc2[nH]ccc12 C(=O)(C(O)CCS(C)=O)NCCN(C(=O)CCCc1nc(C(C)C)no1)CCOC CN1CCC(C(=O)NC2(CNC(c3cc(C4CC4)[nH]n3)=O)CCOC2)CC1=O c1(NC(C=C(C)CN2CCC(Cc3cncc(F)c3)CC2)=O)ccccc1C#N N1(C(CCCCC(C)C)=O)CC(C)OC2(CCN(C(C3CC=CCC3)=O)CC2)C1 N1(C(C2(C=C)CCC2)=O)CC(C2(NC(=O)COCCOCCO)CC2)C1 C1(C(=O)NC(CC)CC)CCOCCC1NC(=O)C(C)OCC1CC1 C(CC(=O)N1CCOC(CC)C1)(C(F)F)NC(CCC(=C)Cl)=O CCC1=C(C(=O)N2CC3CC(O)C2C3NC(=O)C(C)c2ccsn2)CCCO1 C=CC1CN(C(=O)COC(C)CC)CC1NC(=O)Cn1ccc(CC)n1 C(CCCC(=O)N1CC(NC(c2nc(C(F)(F)F)cs2)=O)CC1C)N(C(C)=O)C C(=O)(C1=NOC(C)C1C)N(CCN(C(c1c(C)nc(Cl)cc1)=O)C(C)C)C c1(C(=O)NC2C3CN(C(C=Cc4ccc(C)o4)=O)CC32)csc2c1C(C)CCC2 C1(C(=O)NC(C(N)=O)CO)C2CC3C(C2NC(c2ccccc2F)=O)C13 C(=O)(C(CN(C)C)C(C)C)NCC1C(CC)CCN1C(=O)Cc1ccc(F)cc1 CC(C)C(C)(CNC(c1cc(C2CC2)no1)=O)NC(c1cc(C(F)F)cs1)=O N1(C(c2c(C)cc(C(=O)NC(=O)CC(C)C3CC3)o2)=O)CCCN(C(C)C)CC1 c1(N(C2C3CCC2CNC3)C(C2CNC(=O)O2)=O)ncnc2ccc(F)cc12 CCC(C)C(O)C(=O)N(c1cccc(O)c1F)C(C)(C)C.C12(C)CCCN1OC2=O N1(C(=O)CC2CCN(C(C3(CO)CCOC3)=O)C2)CCC(=C(F)F)CC1 CC(C)(C)C(CO)C(=O)NCC1CCN(C(c2cc(Br)no2)=O)CC1 c1(NC(C)=O)ccc(C)c(C(=O)NCCNC(=O)CS(=O)(=O)CC2CCCO2)c1 N1(C(CS(=O)(=O)N(C)C)=O)CC2(C(=O)NCC3(C)CSC3)CCC1CC2 N1(C(CCC)=O)CCCCC1C(=O)NCCCC(C)NC(c1c[nH]c(=NC)s1)=O N1(C(C(CC(C)(C)C)O)=O)CCC2(CC1)CCN(C(=O)COCP(C)(C)=O)C2 Cn1cc(C(N2CCC(C)(NC(c3c[nH]ccc3=N)=O)C2)=O)n(C)c1=O c1(C(=O)NCC2C(CNC(CNC(C(CC)CC)=O)=O)C2)cc2cc(Cl)ccc2[nH]1 CC(CC(=O)NC1CC2(C1)CC2C(=O)NC1C(O)CC1O)C(F)(F)F C12(C(N(CC(CN(C)C(c3cc(CO)on3)=O)O)C)=O)CCCN1CCC2 Cc1cccnc1NC(c1ccc(CNC(=O)C(c2cn(C)nc2C)O)cc1)=O C#CC1(C(=O)Nc2cn(C)nc2O)CCN(C(=O)C(C)CC=CCC)CC1 c1(C(=O)NC2(CC=C)CN(C(C3(OC)CCC3)=O)C2)c([N+](=O)[O-])cnn1C c1(C(=O)N=c2ncn(Cc3ccncc3)[nH]2)c(Cl)ccc2ccoc12 CC(C)(C)C(C(=O)NCC#CCNC(=O)CC1CCCOC1)N1CCOCC1=O CCCCC(C(=O)N(C1CCN(C(C2CC2C)=O)C1)CC1CC1)C(C)C Cc1cc(C#N)nc(N2CCCC2(C)CNC(=O)C(c2ccc(Cl)cc2)(C)C)n1 N1(C(C(C)OCOC)=O)CCCCCC1C(=O)NCC1CC12CCC2 C=C(C)CCCC(=O)N1CCC(O)(CN(C(c2cccc(C(N)=O)c2)=O)CC)C1 CN1CCN(C(C23CC(CO2)N(N2CC(C=O)C2)C3)=O)CC(O)C1.C(N)=O C1(F)(C(=O)NCC2CCCN(C(CC(CC)OC)=O)C2)CCCCCC1 C(=O)(C(C)CCC(C)(C)C)N1CCC2(CN(C(C3OCCN(CC)C3)=O)C2)C1 c1(C(N2CCOCC(NC(C3CC(C)C3)=O)C2)=O)c(F)ccc(Cl)c1N Cc1cc(OCCC(C)C)ccc1C(=O)NCCC1CC(N)C1(C)C c1(C(=O)NC(C(C)NC(c2nc(C)n(C)c2)=O)(C)C)ncc(Br)cc1F CC1(C)CCCC(O)(C(=O)NC2CCN(c3nc(Cl)ncc3C(N)=O)CC2F)C1 c1(C(=O)NCCCCN(C(c2ccn(CC)n2)=O)C)cc2cc[nH]c(=O)c2s1 c1(C(=O)NC(C)CCNC(C2C3CCCC23)=O)c(Br)sc2ccccc12 C1(CC)(NC(c2cncc(OC)n2)=O)CCCN(C(=O)C(C)OCC2CC2)C1 C1(CC(=O)NC(C(CC)(F)F)(C)C)SC2=NCCN2C1=O Cn1nc(O)cc1C(N1CCC(C(O)CNC(c2cncc(Cl)c2)=O)CC1)=O N1(C(C(c2cnccn2)C)=O)CC2CCC1CC2NC(=O)CN(C)CCO N1(C(c2c(C)nn(CC)c2C)=O)CC2CCN(C(C3C4CC5C(C4)C35)=O)CC12 C1(C(N(CCNC(C(CCC)F)=O)CC)=O)CNC(=O)C(C)(C)C1 N1(C(C2C3CCCOC23)=O)CCC(O)CCCCC1(F)F Cc1cccc(C(N2CCC(O)(CNC(C3CC3c3ccncc3)=O)C2)=O)c1O c1(NC(=O)CC2CC=CCC2)ccc2c(c1)CN(C(c1cccs1)=O)CC2 CN1CCC2(CCN2C(C2(CCNC(C3OC4CCC3C4)=O)CCCC2)=O)C1 N1(C(c2ccn(CCC)n2)=O)CCC(O)(C(C)CNC(c2ccc(Cl)s2)=O)C1 c1(C(=O)NC(CCCC)CNC(=O)CC(C)c2ccco2)ccn(CC)c(=O)c1 C12(C(N(OCC)C)=O)CCN(C(=O)CC3OCCCO3)CCC1C2 C(=O)(CCC(C)O)NCC(C)NC(C1ON=C(C)C1)=O CC12CCC(C1)N(C(=O)C(=O)Nc1cnc(C(F)(F)F)c(C(N)=O)n1)C2 n1(CC(C)O)cc(C(=O)NC2CN(C(C3(C)C=CCC3)=O)CC2C)ccc1=O Cn1ncc2cccc(CCNC(c3nc4cc(F)ccc4s3)=O)c12 C1(NC(c2n(CC)cnn2)=O)CCC2(CC1)CC2NC(=O)C(CC)N1CCCC1 c1(C(N2CC(CN(C(C3C(COC)C3)=O)C)OCC2)=O)ccc([N+](=O)[O-])cn1 c1(CN(CC(N2CC(c3[nH]nnc3C)C2)=O)C)c(C)cc(C)cc1C c1(C(=O)NCC(C)NC(=O)C(C)(C)c2cncnc2)ccnc2ccncc12 N1(C(Cn2ncc(C#C)c2)=O)CC(NC(=O)COCP(C)(C)=O)CC(O)C1 C1(C(N(C2CC2)CC)=O)CCN(C(C2(C)CCSCC2)=O)CC1(C)C C1(C(N2CC(NC(C3C(C)C3)=O)CC(C)(C)C2)=O)COc2cc(Cl)ccc2C1 c1(C(=O)NCCCOCCN(C(=O)C=C2CCCC2)C)coc2ccccc12 CCCCCCC(C)C(=O)NCCC(C)N(C)C(c1ccc(C(N)=O)nc1)=O CCC(C(=O)NCCCC(c1ccccc1)NC(=O)CCCOC)n1ccnc1 CN1CC(N(C(=O)CC23CC(CO2)N(C(c2cnc[nH]c2=N)=O)C3)C)CCC1=O N1(C(c2c(CC)noc2C)=O)CC2CCN(C(=O)CC3CC(C)=NO3)C2C1 c1(C(N(C)CC2N(C(C(CC)O)=O)CCC2)=O)cc(N)cnc1C c1(OC)ccc(CNC(N)=O)cc1C(N1CC(NC(=O)CCSC)C2CC2C1)=O c1(C(=O)NC(CNC(C(C=C=C)C)=O)C)ccc2cnnc(O)c2c1 C(c1ccncc1)=CC(=O)NCCC(=O)NC1CCC(NC(C2CCO2)=O)C1 N1(C(C2N3C(C)CN(CC3)C2)=O)CCC2(CCN(C(=O)C3=COCCC3)C2)C1 C=CC(C)C(=O)N1CC(CN(C)C(c2cc(-c3ccccc3)no2)=O)C1 c1(-c2cccc(C=C)c2)cnn2cc(C(=O)Nc3cccnc3C)cnc12 C1(N(C(C2CCC(=C)CC2)=O)C)CCCN(C(=O)CCOCC2CCCO2)CC1 c1(C(CNC(C(F)=CC)=O)NC(C23CC(CC(C)C)(C2)C3)=O)ccc(C)cc1 CC(O)CCCNC(c1sccc1CNC(=O)C(C)(C)C1CCCC1)=O C(=O)(C1=COCCO1)N1C(CNC(C=C2CCN(C)C2)=O)CCC1 N1(C(=O)Cc2ccccc2O)CCC(F)C(NC(C2(O)CCCCC2)=O)C1 N1(C(=O)NCc2nc(C)oc2)CCN2C(=O)CCC12C c1(CC)cc(C(=O)NCC2CC(O)CN2C(=O)CSc2ccc(Cl)cc2)nn1C N1(C(c2c(C)cccc2)=O)CCCC(CO)(NC(C2CCCN(C)C2)=O)C1 c1(N2CCC3CCN(C(CCC)=O)CC3C2)cc2nc(O)oc2cc1[N+](=O)[O-] CC(C)C(Cc1ccccc1)C(=O)NCC(C)CNC(=O)C(c1cnn(C)c1)=O C=CCCC(F)(F)C(=O)N1CCC(NC(c2cnoc2CC)=O)C(CC)C1 c1(C2C(NC(C(C)NC(N)=O)=O)C2)ccc(Cl)cc1F c1(CC(N2CC3C4CCC(C4)C23)=O)cnn2c1CCCC2 C#CC1CN(C(=O)CC2CC3CCC2O3)CCN1C(=O)CSCC N1(C(C2(OC)CCC23CCC3)=O)CCC2(C1)CN(C(=O)C(C1CCCCC1)O)C2 Cc1cncc(C(=O)NCC(CNC(c2cccc(C(C)(F)F)c2)=O)CO)n1 CC(C)C(C(=O)N1CC2CC1C2NC(=O)CCF)N1CCN(C)CC1 C(=O)(CCC(C)S(C)(=O)=O)NC1CCN(C(c2ccc(C#C)nc2)=O)CC1O C(c1cccc(CO)c1)=CC(N1CC(N(C(C(C)OC(C)(C)C)=O)C)C1)=O C(=O)(CC(O)CNC(=O)Cc1ccoc1)OC.C12(CC1C)C(=O)N2 C1(NC(CSc2nc(C)[nH]n2)=O)CN(C(C2CCC2C)=O)CC12CCCC2 C(=O)(C(O)CC(F)(F)F)NC1(C(=O)O)C2C(C)N(C(c3cc(C)nc(O)n3)=O)C1C2 C(=O)(CC1=CCOCC1)NC(CC)CNC(=O)C(c1ccccc1F)F C1(CN(C)C(C2COCCO2)=O)CCN(C(c2ccsc2Cl)=O)CC1 C1(NC(c2cncc(C)c2)=O)CC2(CCC(CNC(C3CCCCC3)=O)OC2)C1 N1(C(c2c(CNC(c3c(C)ocn3)=O)noc2)=O)CCC2(C)CCCC12 CCCC(C(=O)NC(C)(CNC(=O)Cc1cccnc1C(F)(F)F)CC)OC C(CC(O)CC(=O)NCCN(C(C1CC1C1CCC1)=O)C1CC1)SC C1(C(=O)NCCCN(C(Cc2nc(CC)sc2)=O)C(C)C)CCCSC1C c1(C(N(CCNC(C(CCOC)C)=O)C2CC2)=O)cc(C2CC2)ccc1Cl c1(N(C(C(N2CC(CC)C2)=O)=O)Cc2ccccc2)cnc2c(c1)C(N)CC2 C1(NC(C(C2CCOCC2)C)=O)C2CC(O)C1N(C(c1nccnc1N)=O)C2 C1(C)(NC(C2CCN(CC(C)C)C2)=O)CN(C(C2C(C#N)C2(C)C)=O)C1 CN1CC2CCC1C(NC(=O)C(N1CCC(CCO)CC1)=O)C2 C(=O)(CCSC)N(C(C)COCCNC(=O)C(C)SC(F)(F)F)CC C12(C(N3CCC(C(C)NC(C=Cc4c(C)n[nH]c4)=O)CC3)=O)CCC(CC1)OC2 N1(C(C(CC)CC)=O)CC2CCC(CNC(c3ccccc3F)=O)C2C1 C(=O)(C(=O)C(F)(F)F)NC1CC(NC(C(C)C(C)C2CCCC2)=O)C1 N(C(=NCCF)NCCc1ccnc(Cl)c1)CCNC(c1ccccc1)=O CC(C)CC(C(=O)NC1CCC(NC(C2(c3ccn(C)n3)CC2)=O)CC1)C(N)=O CCCCC(O)C(=O)NCc1cc(C(=O)NOCC(C)C)no1 CC1CCCn2ncc(C(N3CC(N(C)C(c4csc(Cl)n4)=O)C4(CC4)C3)=O)c21 N1(C(C=C(C)C2CC2)=O)CC2CC2(CNC(c2cc(Br)c(Cl)s2)=O)C1 C1(CNC(C(C2CCC2)NC(CSCC(C)C)=O)=O)(CO)CCN(C)C1 N1(C(C(COC)C)=O)CC(NC(=O)CN2C(=O)CCC2=O)C(C2CC2)C1 c1(N2CCN(C(c3nc4ncc(Cl)cc4s3)=O)CC2)cccc2oc(O)nc12 c1(C(=O)NC2C(NC(c3cc(CCC)n(C)n3)=O)CCC2)ccnc(Cl)c1O CC(C)CC(C)C(=O)N1CCCCC1C1CCN(C(=O)CCOC2CC2)C1 c1(OC)ccc(CNC2CC(C(=O)NCCCn3nc(C)nc3C)C2)c(Cl)c1Cl C(=O)(C1CCCc2scnc21)NCCC1(NC(Cc2c(C)nsc2)=O)CCCC1 CCC(C)(C)C(=O)NC1CCCCC1NC(=O)Cn1ccnc1C C1(CCNC(C(COC)O)=O)CCN(C(=O)CNC(c2cnn(C)c2)=O)CC1F CC(C)C(C(=O)NC1CC(NC(c2ccc(-c3ccccc3Cl)o2)=O)C1)N(C)C C1(CCC)(NC(=O)CSC(F)(F)F)CCCN(C(C23CCCC2CCC3)=O)C1 C1(CNC(C2CC2C(F)F)=O)CCCCN1C(c1n[nH]c(C2CC2)n1)=O N=c1[nH][nH]c2cccc(CN3CCC(C(=O)Nc4cccn5nccc45)C3)c12 C#CC1(O)CC(C(N2CC(F)(CNC(=O)CC(C)n3ccc(C)n3)C2)=O)C1 c1(C(=O)NC2CCN(C(c3c(CC)non3)=O)CC2F)cnc2ccc(F)cn12 c1(NC)cnc(C(N2CC(CC(C)NC(=O)Cc3csc(Cl)c3)C2)=O)cn1 C(=O)(CCC(C)C)NC1(NC(C(CC)OC)=O)CCC1.C(CCNC(=O)COC)OC N1(C(C2CC(N(C)C)C2)=O)CCC2CCC(NC(C3CC(C#N)C3)=O)C1C2 N1(C(CCN(C(CCC)C)C)=O)CCCC(N(CCO)C(C2(F)CCC2)=O)C1 c1(COC(c2cc(C(F)F)cs2)=O)cc([N+](=O)[O-])ccc1Cl C1(C(N2CC(CCNC(C3COCCOC3)=O)(OC)C2)=O)CC(=O)OC1(C)C C1(CNC(C2C(OC)C2)=O)COCCN(C(c2cn(C)cc2C(F)(F)F)=O)C1 C(C)(C(=O)N1CCC(CNC(c2cn(C)nn2)=O)C(O)C1)(C(C)C)OC N1(C(C2(CNC(=O)CCc3cnccn3)CCCO2)=O)C2CCCC1CC(O)C2 N1(C(CCC2(C)CC2)=O)CC(CNC(=O)CC2CC(C)(C)CO2)C2CC12 N#Cc1csc(CNC2CCCC2C(N2CC(O)C(O)C2)=O)c1 C1(C(=O)NCC2(C)CC(NC(c3ccc(Cl)cc3)=O)C2)(OC)CS(=O)(=O)C1 CC1CCN(C(C2(C(F)F)CCCO2)=O)CCN1C(C1CC1C(F)F)=O C1(C)(CNC(C2N(C(=O)OC)CSC2)=O)CCC(NC(c2cncnc2)=O)CC1 C1(C(=O)NCC2CCCN(C(c3cc(C)c(Cl)s3)=O)C2)COc2ccccc2O1 CCS(=O)(=O)CC(=O)NC1CCN(C(c2ncc(C)cn2)=O)CC1C(C)C Cc1nnc2n1CC(C(N)=O)N(C(c1ccccc1I)=O)C2.c1cc(O)n[nH]1 c1(CC(C(=O)N(C2CC(C)OC(C)C2)C)N)c[nH]c2cc(F)ccc12 Cc1nc2c(s1)CN(C(=O)C(CNC(=O)C(O)CC(C)C)C(C)C)C2 CC#CCCCC(=O)NC1CCCC(CNC(c2cn(C)c(=O)cn2)=O)C1 C1(CN(C(C2(CCCC)CC2)=O)C)CN(C(=O)C(c2ccccc2)C)CC12CC2 CC(C)C(CNC(=O)CC1NC(=O)NC1=O)C(=O)NCC1(C#N)CCCC1 C1(NC(c2c(-c3ccc(C)s3)c[nH]c2)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1C C(=O)(C1=CC2(CCOCC2)C1)N1CCN(C)C(CNC(C2CC(C3CC3)C2)=O)C1 N1(CC(=O)N(CCNC(c2cscc2C2CC2)=O)CC2CC2)CCCCCC1 c1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CC2)cnn2cccc(C)c12 c1(SC)ccc(C(=O)NC(C)C(CO)NC(C2CCC(F)(F)C2)=O)cc1[N+](=O)[O-] c1(C(=O)NCC2C(CNC(c3cn(C(C)(C)C)nc3)=O)C2)ccc(F)c(N)c1 N1(C(c2c(CC)con2)=O)CCOC(CNC(=O)CCCN(C)C)C1 C(CC(C)C)(C(=O)NCC1CCC(NC(=O)Cc2cnc(C)o2)C1)OC CCCCCCC(=O)N(C(C)CCNC(=O)CCC(=O)N(CC)CC)C(C)C C1(C(=O)O)COCC2(CCN(C(=O)C(c3ccc(F)cn3)(F)F)C2)O1 C=CC1(NC(=O)CC2CCCC2NC(c2ccnn2C)=O)CCCC1 C(=O)(CCC(=O)N(C)CCOCCN(C)C(c1ccnc(Cl)c1)=O)N(C)C C(C(=O)NC(C)(C)CC)(C(C)CC1CCOCC1)N(C)CC1(CC)CCCCC1 C1(NC(CC(C)SC)=O)CC2CCC(C1C)N2C(c1cccc(Cl)c1)=O Cc1nc(C)c(CCNC(=O)C(CCC2CC2)NC(=O)Cc2ccnc(O)c2)s1 CCC(COC)C(=O)NC1C2CC(NC(c3ncccc3N(C)C)=O)CC12 c1(C(=O)NC(c2ccc(OC)cc2)C2CCCC2)ccc(Cl)nc1O C=CCC(C)(C)CC(=O)NCC(C)NC(=O)CCC1CCN(C)C1 Cn1cc([N+](=O)[O-])cc1C(N1CC(CNC(=O)CCS(N)(=O)=O)C(C)(C)C1)=O N1(C(C2(OC)CCCOC2)=O)CC(CNC(C2(C(C)C)CCC2)=O)C(C)(C)C1 N1(C(CC(COC)C)=O)CCN(C(c2ncccc2N=[N+]=[N-])=O)C2COCC12 CC1C(NC(=O)C(C)C(C)(C)C)CC2CCC1N2C(=O)CC1CC(C)(C)CO1 c1(CC(=O)N(C)CC2CN(C(C3OCCN(CC)C3)=O)C2)cc(F)ccc1O C1(CC)CCOCCN1C(=O)C(CNC(c1ccc(=O)n(C)c1)=O)N(C)C N1(C(C(C)(CO)OC)=O)CCCOC(C(N2CCN(C(=O)CNC=O)CC2)=O)C1 c1(C(C)C)ncc(C(=O)N(CC(C)O)CCNC(=O)CC2COC(=O)C2)[nH]1 C1(NC(C(CC=CC)NC(=O)C=CCF)=O)CC2(CCC2)C1OC C(CC1CCCC1)(C(=O)NC(C1CCC1)C1CC1)NC(CSCCC)=O c1(C(C)C)ccccc1OCC(=O)N(CCCN(C)C(c1cn(C)nc1O)=O)C c1(C(CC)CC)nc(Cn2nnc(=O)[nH]2)n(-c2ccc(OC)nc2)n1 c1(C(=O)NCC2C(CNC(CN(C3CC3)CC)=O)C2)cc(F)c2ncccc2c1 C=CC1(CC(N2CC(N3CCN(C(=O)CCOC(C)=O)CC3)C2)=O)CCOCC1 C1(C)(C(=O)NCC(CNC(C2(COC)CC=CC2)=O)(C)O)COC(C)(C)CO1 N1(C(=O)OC(C)(C)C)CCN(c2cncc(NCC3CC(C)CO3)c2)CC1 CN1CCC(C(=O)NCC2(CCNC(=O)CC(C)c3ccccc3)CC2)C1 C1(NC(C2CC(OC)C(OC)C2)=O)CN(C(c2c(C)noc2C)=O)CCC1O N1(C(CC2(COC)CC2)=O)CCC(O)(CCNC(c2cnsc2C)=O)C1 Cc1cccc(C=CC(=O)NC2CCCN(c3cnccn3)C2)c1 CC1CN(C(=O)CCn2cccn2)CC(CCNC(C2CN(C3CCC3)C2)=O)O1 C(=O)(CCC(=O)N1CCCCC1CC(=O)NCC1CC2CCC2C1)NC Cc1nc(NC(C2(CO)CCOCC2)C)cc(N2CCCCC2C2CCC2)n1 c1(OC)cccc(F)c1CN1CCSC(C(=O)N(C2(c3ccccc3)CC2)CC)C1 Cc1c(Cl)nc(CC(C)C)[nH]c1=NCC1CCN(C(=O)C=Cc2nccs2)C1 Cc1cc(NC(C2CC(NC(C3CCO3)=O)C(O)C2)=O)ccc1O c1(C(C)C(=O)NCCC(C)(C)CNC(=O)CC2CCC(O)C2)ccc2c(c1)OCO2 N1(C(c2c(OC)nn(C)c2Br)=O)CC2(CCCCN2C(C2CC2C)=O)C1 C#Cc1ccc(C(N2CC(C(=O)NC(CC)C(F)(F)F)(COC)C2)=O)cc1 C(=O)(C(O)(CN(C)C)C(F)(F)F)NC(C(C)NC(C1CC(F)C(=O)N1)=O)CO N1(C(c2nc(CCCC)sc2)=O)CCCC2(C1)CN(C(=O)CC(C)CF)C2 CN1CCC(NC(=O)C(C2CC2)NC(C2CCS2(=O)=O)=O)CC1=O CCC(C)(CNC(C1CCC(C2CC2)N1C(=O)CCCOCCOC)=O)C(N)=O C1(CC(=O)NC(C)CCCF)(NC(C2COCC2O)=O)CCCCC1 c1(CC)ccnc(C(=O)NC(CC2CCCC2)C(=O)NCC(O)C(C)O)c1 c1(C(=O)NC(CC)CN(C)C(c2coc(C)c2)=O)noc2c1CN(C(C)C)CC2 C1(CNC(CCC#C)=O)CN(C(C2CCCN2Cc2nnn(C)n2)=O)CC12CC2 C1(NC(CCc2ncc(C)[nH]2)=O)CCN(C(=O)C(O)C(F)(F)F)CC12CCC2 c1(NC(c2ccc(Cl)nc2Nc2csnn2)=O)ccc2nccn2c1 C1(C(C)NC(c2cc(C)cc(F)c2)=O)CC2CCC(C1)N2C(=O)CCOC(C)C N1(C(C=C(C)Cl)=O)CCCC(C)(C)C1CNC(C1CC1S(=O)(=O)C(F)F)=O C(c1cnc(OC)nc1)=CC(=O)N(CC(C)NC(c1ncoc1C)=O)CC C1(COC)(CNC(C2CC(F)C2)=O)CCN(C(=O)C=CC2(C)COC2)C1 NS(=O)(=O)C1(C(N2CCN(CCCNC(C3(O)CC(CF)C3)=O)CC2)=O)CC1 C1(C(=O)NCC(CN(C(c2cnc(SC)n2C)=O)C)(C)C)CC2(C1)CC(C)C2 c1(C(N(CC(CC)NC(C2CC(F)(CO)C2)=O)C)=O)c(C)nn(C2CC2)c1Cl c1(NC2(c3n(CCOCC)nnn3)CCSC2C)ccc(OC)cc1CN(C)C C1(C(=O)NCC(C)(C)SC)CCN(C(=O)C=CC2(C)COC2)C(C)C1 C(=O)(CC(C)(C)C)N(CCCC(=O)NCCCOCC(C)C)C c1(CCC)cc(C(=O)NC2CC(F)(CNC(c3sccc3CC#N)=O)C2)n(C)n1 c1(NC(C2CCN(C(=O)CC34CCC(CC3)C4)C2)C)[nH]c(=O)n(C)c(=O)c1C#N c1(C(=O)NC(C(C)NC(c2c(C)nsc2)=O)C(C)C)nccc(N)c1Cl C(c1ccc(C(F)F)cc1)=CC(=O)NCC1C(CNC(C2N(C)CCCC2)=O)C1 N1(N2CC(NC(c3cncc(NC(CC=C)=O)c3)=O)C2)CCS(=O)(=O)CC1 C(C)(C)(CN=c1nc(C#N)[nH]cc1Cl)NC(C(C)CC1CCC1)=O C(=O)(C1=NOC(CN)C1)N1C(C)(CC(=O)NCC23C=CC(CC2)C3)CC1 c12ccoc1C(=O)NC2.C(C(=O)N1CC(NC(=O)N(C)C)C1)(C1(C)CC1)OCC.NC N1(c2nccc(CC#N)n2)CC2CCC(NC(=O)C#CC3CCCCO3)CC2C1 N1(C(C2C(CC)N(C(c3ccc(Cl)c(C#N)c3)=O)CC2)=O)C2CCCC1COC2 C1(C(=O)NC2CC(CC)C2)(CNC(=O)CCN2CCNC2=O)CC(C)(C)C1 C1(CCS(=O)(=O)N(C2C(C)C2)C)CCC2(CC1)CC2 C1(CC(=O)NC(CNC(C(C)(C)CF)=O)C2CCC2)CCOC(C)(C)C1 c1(NC(C)=O)ccc(F)c(NC(C2CC(NC(=O)CC3CC3)CC2O)=O)c1 S(=O)(=O)(c1ccccc1)N(CCC)C(c1ccccc1C(C1CSC1)=O)=O Cc1cc(N2CCC(O)C(F)C2)ncc1S(=O)(=O)NCCc1ncc(F)cc1F Cc1c(C(=O)NC2CCN(C(=O)C=Cc3ccc[nH]3)CC2C)ccc(Br)c1F c1(C(=O)NCC2CC(C)(C)N(C(c3cnsc3)=O)C2)c(N)ccc2nccnc12 N1(C(C(c2c(C)nn(C)c2)C)=O)CC2CCC1C(NC(=O)C(O)CC1CC1)C2 c1(OC)ccc(C(=O)NC2(CCNC(=O)C=CC3CCCO3)CC2)c(F)c1N N1(C(CC(COC)COC)=O)CCc2nc(CNC(=O)C(O)CCSC)sc2C1 CN1CCOCC1C(=O)NCC1CN(C(C2CCC(c3ccccc3)C2)=O)C1 C#Cc1ccc(C(=O)N(C)CCNC(c2cc(-c3ccccc3F)no2)=O)nc1 N1(C(CC(C=C)(C)C)=O)C2CCC1CN(C(=O)C(C)OC1CCCC1)CC2 CC1CCCC1CC(=O)NC1(CNC(=O)CCc2nc(O)n[nH]2)CCCC1 C1(CC)C(=O)NCCCN1C(=O)CC1(NC(=O)C(C)NC(=O)NC)CCCC1 c1(C(=O)NCC2C(C)(C)CN(C(C3(CO)CCCO3)=O)C2)occ2c1CCCC2 N1(C(CSCC#C)=O)CCN(CCNC(=O)COC(C)CC)CC1 O=C(C1=COCCO1)NCCN(C(c1sccc1CO)=O)Cc1cccc(Cl)c1 c1(C(=O)NC(CNC(CCCOCCOC)=O)(C)CO)cccc(N)c1 C1(NC(CC(C)OC)=O)CC2CCC1N2C(c1c(Br)n[nH]c1C)=O CC(C)CC(C)CC(=O)N1CCOC(C(N2CC(C)(CN(C)C)C2)=O)C1 C1(C(=O)N(CC2N(C(CC(C)NC(N)=O)=O)CCC2)C2CC2)CCC(F)(F)C1 C1(N(C)C(=O)C2CC2)CCCN(C(=O)CC2CC23CC3)C1 N1(CCC(=O)NC(C2N(C(CN3C(C)CCC3)=O)CCC2)C)CCCCCC1 C1(C(=O)NC(C(=O)NCC=C)C2CCC2)(COC)CCCOC1 C1(CNC(C2(CC(C)C)CCCC2)=O)CN(C(=O)C=Cc2ncc[nH]2)CC(C)O1 C(C(CC(F)(F)F)NC(=O)Cc1cn(C)nc1C)NC(c1c(OC)cncn1)=O C1(CCC)CCN(C)C(NC(=O)C=C=C(C)C)C1 c1(SC)ccc(-c2nc(CCC(F)(F)F)nn2C(C)C(C)C)cc1 C(N=c1[nH]c2ccc(O)cc2s1)C1CCCC(NC(CCc2n(C)cnc2)=O)C1 C=CCCCC(C(=O)N1CCC(F)(CF)C1)NC(=O)CSC CC(C)CCC(=O)N1CCC(N(CCO)C(c2ccc(-c3cccs3)s2)=O)C1 c1(C(N2CC(C(=O)Nc3c(CC)ncc(Br)c3)C2)=O)c(Cl)cnc(Cl)c1Cl n1(CCC(=O)N(CC(CN(C(=O)C=Cc2ncc[nH]2)C)O)C)ncn(C)c1=O C1(NC(c2c(Cl)cn(C(C)(C)C)n2)=O)CC2CCC(C1)N2C(C1CCCOC1)=O N1(C(=O)OC(C)(C)C)C(NCCC[SH](c2ccn(CC)n2)N)CCC1C1CC1 C1(C(C)(C)O)CCN(C(C2CCCC2NC(=O)CC#N)=O)C1 c1(OC(C)(C)C)cc(F)cc(C(=O)NC2(n3cnnn3)CC2)c1N c1(CC)cc(C(=O)NCC2CC(C(F)(F)F)CO2)cc(C)n1 Cc1nccc(C(=O)NCC2CCCC2C(N2CC(CCO)C2)=O)c1N C1(c2n(CCC)nnn2)(Nc2cnn(C(C)C)c2C)CC(C2CC2)(C2CC2)C1 CC(C)C(C)(CNC(C1CC1(F)F)=O)NC(c1ccc(-c2ccccc2)n1C)=O N1(C(C(C=C)O)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)OC2(CCC2)C1 c1(CC)n[nH]cc1C(N1CCC(C(N)=O)C1)=O.c12ncoc1CNC2=O C(=O)(CCC(CC)OC)N1CC(NC(c2c(CC)noc2C)=O)C(O)C1 Cc1cccc2[nH]cc(C(N3CCCC3(C)CNC(C3CCN(C)C3=O)=O)=O)c12 c1(OC)cccc2c(=O)c(C(=O)NC3CCC(NC(C4CCCO4)=O)C3)c[nH]c12 C1(CCCC)CCCCN1CC(=O)NC1(c2ccc(OC)cc2)CC1(C)C c1(OC)ccccc1SCC(=O)NCC1CCCN1C(=O)C(C)(C)c1cnsc1 C1(CC(=O)N(C(C)CNC(=O)C(C)S(C)(=O)=O)C)CCC2(CCC2)CO1 c1(C(=O)NCC(C2CC2)NC(c2cnccn2)=O)csc(Cc2cnn[nH]2)n1 C(=O)(CP(=O)(C(C)C)C(C)C)N1CC(CNC(C=CCCC(C)C)=O)C(O)C1 C#CC1(C(=O)NCC(c2nccs2)C)CN(C(=O)CC2C=CCC2)C1 c1(C(N2CCC(CCNC(C(C)SCC)=O)C2)=O)cc(N(C)C)ncn1 C(F)(F)(C(F)(F)C(F)(F)F)OCC(N1CCC(NC(c2ccncc2Cl)=O)C1)=O C1(NC(c2cc(C)cc(F)c2)=O)CC2CCC1CN2C(c1csc(C)c1C)=O c1(CC(=O)NCCN(C(CC=CC)=O)C)cc(C)no1 c1(NC(C2CCCN(C(=O)NCC(N3CCCC3)C)C2)=O)cccc(=O)n1C c1(C(=O)NCC(C)CNC(C2CCC2)=O)cc2c(cc1Br)OCO2 N12CC3CC(C3C1)SCC2=O.C1(=O)C(C)N1.C(=O)(NCC)NCC c1(C(N(CCCNC(C2CC2C2CCCO2)=O)CC)=O)ccoc1Br c1(OC)ccc(-c2ccccc2C(F)F)c(C)c1C(=O)OC N1(C(c2nc(CC)sc2)=O)CC(CNC(=O)C(C)CN(C)C)OC(C)(C)C1 N1(C(C2(C=C)CC2)=O)CCCN(C(=O)CSCc2cscn2)CC1 C(=O)(C(O)P(C)(C)=O)NCC(C)(C1CC1)NC(CC(n1c(CC)ncc1)C)=O C1(C2CC2)(NC(Cc2nc(CC)sc2)=O)CCN(C(=O)CC2CC3(CC3)C2)C1 N1(C(CC=CCC)=O)CC(F)(CNC(c2cnn(C3CCCCC3)c2)=O)C1 N1(C(C=CC=CC)=O)CCC(C2CCN(C(c3cccn4nnnc34)=O)CC2)C1 C(CCCOC)(C(=O)NC1CCCC(O)CC1)NC(C(CC)CN(C)C)=O c1(C(C(=O)NC2CC2CNC(C2C=CCS2)=O)OC(C)=O)ccccc1 C1(CNC(=O)OC(C)(C)C)CCCCC1C(N1CCC(C(N)=O)C1)=O C12(NC(C3ON=C(CC)C3)=O)CCC(C1)N(C(=O)C=Cc1cscn1)C2 C(=O)(CCCCC(C)C)NC1C(OC)CN(C(=O)CN2CSCC2=O)C1 N1(C(C2C(C(C)NC(c3cnc(O)n3C)=O)C2)=O)CCC(CF)CC1 Cc1c(Cl)ccc(C(=O)NC23CCC(C2)N(C(c2cncn(C)c2=O)=O)C3)c1O C(=O)(CCCC1CCCO1)N(C1CN(C(=O)C(C2CCOCC2)O)C1)C CN1CC=C(CC(=O)NC2CCCCC2C(=O)N(C)Cc2ccns2)CC1 C(=O)(C(C(CC)CC(C)C)N1CCCC1CC(C)C)NCC=C N1(C(C2C(C#N)C2)=O)CC2(NC(C3CCN(c4ccncc4)C3)=O)CCC1C2 C1(C)(C(N(C(C)C)CCN(C)C(C23COC(CF)(C2)C3)=O)=O)CCCCCC1 Nc1ccc(Br)cc1C(N1CCC(CF)(NC(=O)CCc2cnc[nH]2)C1)=O CC1CCCN(C(C2CCCN2C(=O)OC(C)(C)C)=O)CC1.C12(CC1C)C(=O)N2 Cc1c(Cl)ccnc1C(N1CC(=C(F)CNC(C2CCc3nc[nH]c3C2)=O)C1)=O N1(C(CCN(C(=O)C(C)CN=[N+]=[N-])CC)=O)CCc2c(nnn2C)C1 c1(OC)cccc(C(N2CC(CNC(c3snnc3C(C)C)=O)CC2C)=O)c1N C1(CCC(=O)N(CC)Cc2csc(C)n2)CCN(C(C2CCNC2=O)=O)CC1 Cc1nc(NCC2CCCCC2C)cc(N2CCNC(=O)CC2)n1 C1(C(=O)NC2CCC(N(C)CC)C2)COCCC1NC(=O)CC1CC1OC CS(=O)(=O)CCCC(=O)N1CC2CCCC2(CNC(c2cc3cscc3s2)=O)C1 c1(OC)noc(C(=O)NC(CNC(c2ccn(C3CC3)n2)=O)C2CC2)c1Br CC1(C)CC(C(=O)NCCC2CC(F)C2)CCN1C(c1cc(C#N)c[nH]1)=O C1(C(N(C)CCOCCNC(=O)Cc2cn(C)nn2)=O)COCC(C)(C)O1 CC(C)(C(=O)N1CCC(C(=O)NON2CCC2CO)C1)c1csc(C(F)(F)F)n1 c1(C(N(CCCN(C(c2cc(C(C)C)on2)=O)C)C)=O)cc2cccnn2c1 c1(C(N2C(C)CC(NC(C3(C=C)CC3)=O)C2)=O)ccc2cccc(Cl)c2n1 C12(C(=O)Nc3c(OC)cccc3Cl)CCN(C(=O)C(F)C(F)(F)F)CCC1C2 N1(C(c2cc(C(C)C)nn2C)=O)CC2CCC2(CCNC(=O)CSC2CC2)C1 C(=O)(C(C(C)(C)C)NC(N)=O)NCCC(C)N(C(=O)CSc1ccc(Cl)cc1)C CC1CN2CCN1C(C(=O)NCCCN(C(=O)C(C)(F)C(F)(F)F)C1CC1)C2 N1(C(c2ccnc(C)c2N)=O)CC(CNC(c2ccoc2Cl)=O)OC2(CCC2)C1 C12(C(=O)NCc3c(C(=O)NC(CC(=O)OC)C)con3)CCC(CC1F)C2 N1(C(c2cc(C)no2)=O)CCCC2(CNC(C3CCCC3)=O)CC12 C12(C(=O)NCC(C)C3CCC3)C(NC(c3cnco3)=O)C3CC1C2C3 C1(CC)CN(C(=O)CCC(C)(F)F)CCN1C(c1ccnn1CC)=O C1(CNC(CNC(=O)OC)=O)CN(C(C2CC3(C2)CC(O)C3)=O)CCCO1 CON(CCC(=O)N1CCCC(C)(O)CC1)C(=O)C(C)n1ccnn1 C12(NC(C=C(CC)CC)=O)CCOC(CNC(=O)C(c3ccc(F)cc3)O)(C1)C2 C1(CCNC(COC(C)C)=O)CCN(C(C2CCCC(=O)O2)=O)CC1 C1(CNC(c2c(CC)ocn2)=O)CC12CCN(C(c1cncc(Cl)c1Cl)=O)CC2 CC(CCNC(=O)C(O)C1CC1)NC(N)=O.C1(=O)C(=O)NCCN1 C(c1cc2ccccc2n1C)=CC(=O)NCC(C)N(C(c1c(CC)nns1)=O)C C(=O)(C1SCCc2sccc21)NCC(C1CCC1)NC(C(COC)(C)C)=O CC1C(=O)NCCN1C(=O)CCCC1(NC(c2cc(F)cnc2O)=O)CCC1 c1(C(=O)NCC2C(NC(COC(CC)C)=O)CCC2)ccc(Cl)c(F)c1 c1(C(N2C(C)CN(C(CCCCCC)=O)C(C)C2)=O)cc(N)c2ncccc2c1 N1(C(C2(C)CC(F)C2)=O)CCC(C2CCCN(C(C34CCCCC3C4)=O)C2)C1 Cc1cc(C(=O)NC(C)C(=O)NCC2CN(C)CCO2)ncc1N N(C(=NCCC1=CCOCC1)NCC(F)F)C(c1ccc(F)c(Cl)c1)C N1(C(c2c(CC)cccc2)=O)CCN(C(c2cc(SC)oc2C)=O)C(CO)C1 C(C1=NOC2(CCC2)C1)NC(C1(C#C)CCN(C(=O)C(C)OC)C1)=O C1(c2ccccc2)(C(=O)Nc2ccc(-c3nn[nH]n3)o2)CCCO1 Cc1ccc2nc(NC(C3CC(NC(=O)CC4CC5CC5C4)C3)=O)cn2c1 c1(C(C)=O)cc(C(N2CC(CNC(=O)CN(C)C(C)C)C2)=O)ccc1F N1(C(C2(CC)CCOCC2)=O)CC2CN(c3ncnc(=N)[nH]3)CC2C1 C1(C(=O)NCC(c2c(C)cccc2)O)CC12CCS(=O)(=O)CC2 C(=O)(CS(=O)(=O)CCOC)N(C1CCN(C(CSCC(=O)OCC)=O)C1)C N1(C(CNC(C2CCN(CCN3CCCCC3)CC2)=O)=O)CCCC(C#N)C1.CS c1(-c2ccn(C)n2)nc(CCc2ccc(F)cc2)n(C2CCS(=O)(=O)C2)n1 N1(C(CC2CN(C(COCC(=O)NC)=O)CC2C)=O)CCC2(CC(CO)C2)C1 N1(C(CC2(C)CC2(Cl)Cl)=O)CCC2(CC1)CC2CNC(=O)CCCN=[N+]=[N-] N1(C(CC(c2c(OCC)cccc2)NC(C)=O)=O)CC2CCCC1C2 c1(C(=O)NCC2N(C(C(C)CC3CC3)=O)CC2)ccc(F)c2[nH]ccc12 C1(CC=C)(NC(c2coc(C3CC3)n2)=O)CCN(C(=O)CCC2CCCOC2)C1 C(CC(C)(C)CC(=O)NC(C)CN(C)C(c1cncc(C(F)F)c1)=O)OC c1(OC)ccc(-n2cc(C(=O)NC(C)(C)C)nn2)cc1.N1(C(=O)O)CC(CO)CC1CO Cc1cccn2ncc(C(N3CCCN(Cc4ccc(CO)c(Cl)c4)CC3)=O)c12 c1(CCC=CC(=O)NCC(C)N(C(=O)CC2CCCC2)CCOC)ccccc1 Cc1cc(C(=O)NC2CN(C(=O)CNC(c3ccsc3)=O)CCC2C)ccc1O c1(C(N2CCCC(C)C2CNC(=O)CC#N)=O)c2c(nn1C)CCSC2 N1(C(C2(C)C(C)(C)C2)=O)CCCC2(C1)CN(C(c1cnn(C3CCC3)c1)=O)C2 c1(C(=O)NCC(CO)NC(C2(Cl)CC2(F)F)=O)cncc2c(O)nccc12 CC(O)C(C(=O)OC(C)(C)C)NCc1c(Br)cnn1C.N1(C)CCN(C(=O)N)CC1 C1(C(=O)NC2CC(CNC(c3c(C(C)C)noc3)=O)C2)CC(O)CN1C(N)=O N1(C(C(C)S(N)(=O)=O)=O)CCCC2(CCN(c3cncc(C#N)n3)C2)C1 c1(C(C)(C)CNC(c2cncs2)=O)cccc(Cl)c1F.C12CCCCN1C(=O)C2 Cc1nn(C)c(=O)c(C(N2CCN(C(c3ccc(N)cn3)=O)C(C)C2)=O)c1C Cc1cc(-c2noc(-c3ccc(N4CC(C)OC(C)C4)nc3)n2)c(N)cc1F C1(NC(Cc2cc(C)no2)=O)CCCCC12CCN(C(c1ccc(Cl)o1)=O)C2 C1(COC(CCC#CC)=O)CCC(C)CN1C(=O)OC(C)(C)C c1(CC)cc(C(=O)NCCCOCCN(C)C(C2NC(=O)CC2C)=O)cc(N)c1 CC(CC(C)(F)F)C(=O)NC1CCN(C(c2ccccc2CO)=O)CC(O)C1 Cc1nc(C(F)(F)F)c(NC(C2CN(Cc3cn(C)nn3)CCO2)=O)s1 CC1CC(NC(=O)C=CCN(C)C)CN1C(c1csc(-c2ccoc2)n1)=O CC1(C)C(NC(C2CCOC2CNC(c2cc(CO)on2)=O)=O)C1(C)C c1(C(=O)NCCC(=C)CNC(=O)C(C2CCOC2)OC)cn2cc(Cl)cnc2n1 C1(C(N2CCN(C(C3CCCO3)=O)C(CC(F)F)C2)=O)CCc2c[nH]nc2C1 CC(O)C(F)(F)C(=O)NC1(C)CCC(NC(=O)CCOc2cccnc2)CC1 N1(C(C(CCC)N(C)C)=O)C2CCC1CN(C(c1ccc(C)nn1)=O)CC2 c1(C(C)C)cncc(C(=O)NC2CC(CNC(c3cnc(C#N)s3)=O)C2(C)C)c1 N1(C(=O)CC2CCC(O)C2)CCC2(CCCN2C(c2ccc3nccn3n2)=O)C1 C(=O)(CC(F)F)NC(C1CCCN1C(=O)CCc1cnc(-c2ccccc2)o1)C C(c1ccccc1F)=CCC(=O)N(CC(C)O)CCNC(C(C=C)OC)=O Cc1nc(C(=O)NCCC2(CNC(=O)COc3ccon3)CC2)cc(O)n1 C1(c2nnnn2CCSC)(Nc2cccc(OC(CC)(C)C)c2)CCC(C)SC1 C#CCC(C(=O)NC(C)C(C)(C)CN(C)C)NC(c1nc(Cl)oc1C)=O c1(OCCN(S(C)(=O)=O)C)ccc(OCCO)cc1.c12ccc(cc1)CN2 C#CC1(NC(C2CC(=C)CCN2C(c2ccc(F)s2)=O)=O)CC2CCCC12 C(N=c1nc(Cl)[nH]c(OC)c1C#N)C1CC(NC(c2c(CC)occ2)=O)C1 C1(NC(C(C)(C)OCC)=O)C2CC(CN(C(c3c[nH]nc3C(C)C)=O)C2)C1CO n1(CCN(C(=O)C(c2cc(F)ccc2F)CN)C)cnc2ccccc12 c1(C(N(CCC(C)NC(C2(S(N)(=O)=O)CCC2)=O)C)=O)ccn2ncnc2c1 C(=O)(C(O)CC1CCCC1)NCCCN(C(=O)CC1(C2CC2)CC1)CC C(C1CCCCCC1)=CC(=O)NCC(=C1CN(C(C2C3CC4C(C3)C24)=O)C1)F c1(-c2nc(C(CC)O)nn2CC(C)(C)C)cnc2c(c1)CCOC2 CC(C)CCC(=O)N1CC(OC2C=CCN(C(=O)C=CSc3ccccc3)C2)C1 C1(C(=O)NC2(CCNC(C(CCSC)O)=O)CC2)CCCNS1(=O)=O C1(SCCNC(C(C2(C)CC2)NC(C)=O)=O)CC(C)(C)C1 n1(CCC#C)c(N2CCN(C(c3ccccc3)C)CC2)nnc1-c1cccn1C N1(CC)CCCC(C(=O)NC2CCN(C(=O)CCC(=O)N(C)C)C2CC)C1 N1(C(CCOc2ccc(C)cc2)=O)CC2(CC(CNC(C3(C)CC3(F)F)=O)C2)C1 N1(C(C=CCC)=O)CCC(C)(NC(C2CCC(=O)N(c3cnn(C)c3)C2)=O)CC1 c1(C(=O)NCC(C)N(C(CNC(C)=O)=O)C)ccccc1C#CC1CC1 CC12CC(C(=O)NCC(C3CC3)NC(C3CC4C=CC3C4)=O)(C1)C(C)(C)O2 C1(NC(C2C(OC)CCCC2)=O)(CO)CCN(C(=O)CC2(C(F)(F)F)CC2)CC1 Nc1cc(C(=O)NC2CCC2CNC(c2csnn2)=O)nc2ccccc12 c1(C(N(C2CCN(C(Cn3ccc(C)n3)=O)CC2)C)=O)cnc2n1CC(C)CC2 C=C(C)CCCC(=O)N1CCCCC1C(=O)NCCNC(=O)NC(C)C Cc1ccc(CNC(=O)C(O)C2CN(C(c3n[nH]cc3C)=O)C2)cc1 c1(C(N(CCCN(C(C(C#C)(C)C)=O)C)C)=O)cc2cc(C(F)(F)F)ccc2s1 C12(NC(C(CC)O)=O)CCOCC1CN(C(=O)CS(=O)(=O)NC(C)(C)C)C2 C(=O)(CC(C)NC(=O)C(C1CC(NC(c2cnn(C(F)F)c2)=O)C1)OC)OCC N1(C(CCc2cc(C)on2)=O)CCCCC(CNC(=O)CSc2ccccn2)C1 N1(C(c2ncc(C(=O)OC)s2)=O)CCN(C(=O)C(C)NCC2(CSC)CC2)CC1 C1(CN(C(CN(C(=O)OC)C)=O)C)CCCN1C(=O)CN1CC2CC2C1 C12(C(=O)NC(C)CCNC(=O)C=CCO)CC(N=[N+]=[N-])C1C2 N1(C(C2(CC=C)CC2)=O)CC2CC2(NC(c2scnc2C(C)C)=O)C1 C(C(F)(C(=O)N1CC2(CCC(=O)O2)C1)C(C)C)NC(c1cc(C)c(O)nn1)=O N1(C(c2nnc(C)s2)=O)CCOC(CC(=O)Nc2nccnc2Cl)C1 CC1CCOCC1C(=O)NCC1(F)CC(CNC(c2cc(Cl)no2)=O)C1 C1(C(N2CC(NC(CCC(CC)OC)=O)C2)=O)CCn2ccnc2C1 CC1CCCC(C(=O)NC(CC(=O)NCC2COC(=O)N2)C(F)F)CC1 c1(C(N2C(CNC(c3c(C)con3)=O)C(C)CC2)=O)ccc2c(c1)COB2O c1(C(=O)NC(CCOC)CNC(c2ccc(=O)oc2)=O)cnn2c(C)ccnc12 c1(OC)cc(CNCC2COCCN2C(c2cnon2)=O)c(Br)cc1O c1(OC)cc(C)cc(C(=O)N(C(C)CC(c2c[nH]c3ccccc23)=O)C)c1C N1(C(C2CCCS(=O)(=O)N2)=O)CCN(C(=O)CSCC(F)F)C2(CCC2)C1 Cc1ccc2c(C(=O)Nc3cc(C4CC4)cc([N+](=O)[O-])c3)csc2c1 C(=O)(C(O)CCC(C)C)N1CCCN(C(c2n[nH]c(C)c2C)=O)CC1 N1(C(C(C)=CC)=O)CCN(C(C23CCC2CC3)=O)C(CCCC)C1 CCCCC(C(=O)N1CCC(CO)(CNC(=O)CCCC(C)=O)CC1)N(C)C CC1CCCC(N=c2[nH]c(=NCCNC=O)c3[nH]ccc3[nH]2)C1 N1(C(C(CC(C)C)NC(c2ccc(C(C)N(C)C)o2)=O)=O)CCc2sccc2C1 c1(C(=O)NCC(CC(=O)N(CCOCCOC)C)O)ccc2cc[nH]c2n1 N1(CC(N2CC(OC)(CNC(=O)C(F)(F)CO)C2)=O)CCCCC(O)C1=O C=CCC(F)(F)CNC(=O)NCc1ccc(NC)cc1 C(=O)CCCCC(F)(F)F.C1(c2cn(C3C(C)CNC3)nn2)CC2CCC1CC2 c1(C(=O)NCC(=C)CCNC(=O)COC(CC)CC)ccccc1SC1CC1 Cc1nc(NC2CC(CNC(C3CCC4(CC4)C3)=O)C2)cc(SC(C)C)n1 N12CCC3(CC1)CC3(C)C(=O)N1CCC(CCO1)CCC(CCCC)(CC)C2=O N1(CC)C2CCC1CN(C(=O)C(C)(C)C(C)NC(c1ccc(N)cn1)=O)C2 c1(C(N2CCC(CCC)(NC(c3cnco3)=O)CC2)=O)ccc([N+](=O)[O-])cc1O CC(C)CCCCCC(=O)NC1CCCN(C(c2cc(F)cc(Cl)c2)=O)C1C C1(C(=O)NC(C)CNC(C2CC(c3cccc(F)c3)(F)C2)=O)(CC)CCCCC1 C12CCC(CC1)CC(=O)NC2.c1(CNC(C2(C(=O)OC)CC2)=O)cnc(SC)o1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NC(CNC(C1CC1C#N)=O)C(C)(C)C N1(C(C(=O)Nc2c(OC)cccc2)C2CC2(C)C)CCCc2c1ccc(C)c2F N1(C(Cc2nc(C)oc2)=O)CCC2(CC1)CC2NC(=O)CCCN1CCCC1 c1(NCCNC(=O)Nc2ncc(C)cc2Br)ccc(F)c2ccccc12 C1(C(=O)NCCN(C(c2ccon2)=O)C2CC2)CC12CCC1(CC2)OCCO1 N1(C(C(C2CCC2)OC)=O)CCC(C2CC2)C1CNC(c1ccc(=O)n(O)c1)=O C1(NC(C(C)SC(F)(F)F)=O)CCN(C(c2ncccn2)=O)C(C)C1 c1(C(N2CCN(C(C3CC3(F)Cl)=O)CC2)=O)cc2cc(Cl)sc2[nH]1 C1(C(F)F)(CNC(c2c(C)scn2)=O)CCN(C(C2CCS2(=O)=O)=O)C1 c1(C(=O)NCC2(NC(C3(SC4CC4)CC3)=O)CCOC2)cc2ccccc2[nH]1 N1(C(c2n(CC)ncn2)=O)CCC(CNC(=O)C(C)(C)N2CCCC2)C1(C)C CC1(C)CCC(C(=O)Nc2cc(C#N)ccc2F)CN1C(=O)C=CC1CCOC1 N1(C(c2c(C(N)=O)csc2)=O)CC2(CCC(NC(c3cnccc3Cl)=O)CC2)C1 c1(CCC)n[nH]c(=NCC(c2ccccc2F)NC(=O)C2CC2)s1 N1(C(C(C)NC(C)=O)=O)CCC(CCCNc2ccccc2OC(C)C)CC1 C(=O)(C(F)CC(CC)CC)NC(CCC)C(=O)NCCOC1(C)CCCC1 C1(N(C(C(C=C)O)=O)C)CN(C(=O)C#CC2(C)CC2)CC12CC2 C1(NC(C2(C)COC2)=O)CCC(NC(C2CCC(F)C2)=O)CC1 N1(S(C(C)C)(=O)=O)CC2CCCC1C2C(=O)NC12CC(c3ccccc3)(C1)C2 Cc1nn(C)c(C)c1NC(C12CC1CCC2NC(=O)CN(C)C(=O)OC(C)(C)C)=O CCCC(CCC)C(=O)NCCC1(CNC(C2CCNC2=O)=O)CC1 c1(C(N(C)CC2N(C(c3cc(CC)on3)=O)CCC2)=O)ccc(C)nn1 N1(C(C2OCC(C)(C)C2)=O)CCCC(C(=O)NCCN2CCC(F)(F)C2)CC1 c1(CC)ccc(CCC(=O)NCC(C)CN(C)C(c2c[nH]nc2C(C)C)=O)cc1 c1(CNC(C(c2cn(CCO)nn2)NC(CC=C(C)C)=O)=O)ccc(F)cc1 c1(CCC(=O)N(C(CNC(CC(C)N2CCCC2=O)=O)C)C)cc(F)cc(F)c1 CC1CC(NC(=O)C(F)OC(F)(F)F)CCN1C(c1cc(N)ccc1F)=O C1(N(C(C2(OC(C)C)CCC2)=O)CC)CCCN(C(=O)Cn2c(C)csc2=O)C1 c1(C(N2CCC(C)(CNC(COCCC)=O)C2)=O)cscc1S(C)(=O)=O CC1=C(C(=O)N(C2CCCC2)CCNC(C2CC23CCCOC3)=O)CCC1 C(=O)(C(C(C)NS(=O)(=O)c1cccnc1)C(C)C)NCc1ccc(COC)cc1 C1(NC(c2nc(C)c(C)[nH]2)=O)CCN(C(=O)CCOC(C)CC(C)C)C(C)C1 C1(C2CN(C(C3COCCO3)=O)C2)(NC(CC(=O)OC)=O)CC1 C(=O)(C1=CCC(C)CC1)NCC1C(C)CN(C(=O)Cn2cncn2)C1 c1(OC)cc(C(=O)NCCC2(CNC(c3csc4cncn34)=O)CC2)c(Cl)cn1 C(=O)(CC(=O)N(CCCN(C(=O)C(CC)c1cccnc1)C)C)NCC C=CCCC(CC(C)C)C(=O)N(CCCNC(c1ccc(C2CC2)o1)=O)C1CC1 C#CCC(C)(C(=O)NCC(=O)N(C)OCC)NC(=O)Cc1nocc1C CCCC(C(=O)NCC1CCC1NC(=O)C=C1CN2CCC1CC2)C(C)C c1(CNC(C2CC(F)CN(Cc3cc(C)ncc3)C2)=O)cnc2[nH]ccc2c1 C1(NC(C(COC)(F)F)=O)CCCCC1NC(c1cc(CO)oc1C)=O.S(C)(=O)(=O)N c1(SC)cc(C(=O)N(C(CNC(C2(SC)CCCCC2)=O)C2CC2)C)ccn1 c1(C(=O)NC(CSCC)C(=O)NCC2CCC3CC23)csnc1Cl C1(CNC(CC)(C)C2CC2)CCC2(C1)OCCO2 C(CC(C)(C)C(=O)NO)O.C1(OC)CCCC(C(=O)NCCC(=O)N(C)C)C1 C1(NCc2ncc(C)[nH]2)CCc2nc(C(=O)O)cn2C1 C1(C)(C(=O)NC(c2scc(C)n2)CO)CCCN(C(c2cnn(CCN)c2)=O)C1 c1(C(=O)NCC2C(NC(C(CCCOC)C)=O)C2)cc2oc(Cl)cc2[nH]1 C1(CNC(c2c(SC)cn(C)n2)=O)CN(C(C2(CO)CC(F)(F)C2)=O)CCN1C Cc1cc(C(=O)NCCC2(O)CN(C(=O)C(c3ccc(Cl)s3)C)C2)on1 C=CCCC(C(=O)OC)NC(C1CN(C(=O)C(F)C(F)(F)F)CC(C)O1)=O c1ccc2cc(CNC(c3ccn(C4CC4)n3)c3nnnn3C3CC3)ccc2c1 C(c1ccc(F)cc1F)=CC(N1CCC(NC(=O)Cc2cnc[nH]2)C1C1CC1)=O N1(C(C(CC)O)=O)CC2(CCC2)CCC1CNC(=O)C(C)CC1CCC1 c1(C(=O)NC2CN(C(CCSCC)=O)CC2F)ccc(F)c2cccnc12 c1(CN2CC(C)(C)N(CC(c3ccsc3)O)CC2)ccc2c(c1)CCC(=O)N2 N1(CCNC(C)=O)CCC(=O)N(Cc2nnc(-c3cccc4c3OCO4)s2)CC1 c1(C(CNC(C2CC(O)C2)=O)NC(C(C)(C)OC(C)C)=O)ccc(Cl)cc1 N12CCc3ncc(n3CC1)NC2=O.c1(CNC(=O)OC)ncccc1C(F)(F)F c1(CN(C(c2ncc(Cl)n2C)C(=O)NCC(C)C)C)cc(F)ccc1F c1(N2CC(CNC(CCC)=O)(OC)C2)ncnc2sc3ccccc3c12 C(=O)(C(C(C)(C)C)C1CCCC1)NC(CNC(c1c(OC)ccnc1)=O)C(C)C CC1CN(C(c2cc(F)cnc2N(C)C)=O)CCC1NCc1ccccc1 C1(CC(N2CCC(C)(C)C2)=O)CN(C(=O)CC2CC(F)(F)C2)CC12CC2 C1(NC(c2cnn(-c3ccccn3)c2)=O)CCCCC1NC(c1csc(O)n1)=O c1(C(=O)OC)cc(C(N2CCC(CCNC(=O)CCOC3CCC3)C2)=O)on1 C(C(=O)N1CCCC1CF)(C(C)(C)C)OC.c1(N2CCC2=O)cccc(F)c1F c1(OC)cc(NC(C)=O)ccc1OCC(N1CC2CN(c3ccccc3)C2C1)=O C1(NC(CCc2onc(CCC)n2)=O)(CO)CCN(C(C2CCCN2N=O)=O)C1 C1(CCNC(c2cnc(C(F)(F)F)cn2)=O)COCCN1C(C1SCCS1)=O C1(CC(=O)NCC2CC(NC(CCN(C(CCC)C)C)=O)C2)CC(=O)NC1=O C1(C(C)(C)O)CCCN(C(C2COCCN2C(c2cscc2Cl)=O)=O)C1 C1(NC(CC(C)C(F)F)=O)CCN(C(=O)CC(=O)NCC2CC2)C12CCC2 N1(C(C(CC)NC(C)=O)=O)CCC(CNC(c2cnc(C3CCC3)o2)=O)CC1C CCC(CC(=O)NCC1CCC(C(=O)N(C2CCC(C)(C)C2)C)C1)C(C)C CCS(=O)CC(=O)NC(C)(C)CCC1CCN(C(c2cc[nH]c2)=O)CC1 C1(CNC(c2cc(C(C)C)on2)=O)CCN(C(=O)C(F)n2cccn2)CC1C CC(C)C(C)CC(=O)N(C1CN(C(C2(C(F)(F)F)CCC2)=O)CCC1C)C C1(CNC(C(C)(C)COCC(F)F)=O)CC12CCN(C(c1n[nH]cc1F)=O)CC2 c1(C(=O)NCC(C)N(C(=O)C(C(C)O)N(C)C)C)cc(F)ccc1F C(CC(C(=O)NCCCN(C)C(C1(CCOC)CC1)=O)NC)SC.c1(C)ccccc1 c1(C(N(C2CN(C(c3c(C)cc[nH]c3=N)=O)CC2F)C)=O)ccc2cncn2c1 N1(C(C(COC)O)=O)CCC2(CCCCN(C(=O)C=CC3CCCO3)C2)C1 C1(NC(c2n(CC#C)ccc2)=O)CC2(CCN(C(=O)CCC)CC2)C1 C(c1cc2ccccc2o1)=CC(N1CCC(O)(C(C)NC(=O)C(C)C#N)CC1)=O C12(C(=O)NC(C3(C(=O)NCC4CC4)CC3)C)CC(C1)C(C(F)(F)F)O2 C1(C(=O)NC(c2ccnc(C)n2)C)CCC2CCC1N2C(c1cn(C)cc1C)=O CC1CCN(C(=NCCC2CCSC2)NCC(CC2CCC2)CO)CC1 O=S(=O)(c1ccc(N2CCC(F)(CO)CC2)cc1Cl)N1CC2(CO)CCC1CC2 C(=O)(C#CC1(C)COC1)NC(C(=O)NC(C1CCCCC1)C)C1CC1 c1(SC)cc(CNC(=O)Nc2nc(C(C)(F)F)cs2)ncc1F N1(C(CN(C)CC)=O)CCC(NC(C2(C(=O)NC3CC3)CC2)=O)C1.C1CCC1 N1(C(C(C)N(CC)CC)=O)CCCC2(CCN(C(=O)C(C(C)C)N(C)C)C2)C1 C(=O)(CCS(=O)(=O)C(F)(F)F)NC1CC(N(C(CN2C(C)CC2)=O)C)C1 c1(CCC(=O)NCC(CNC(C2C(C3C(C)C3)C2)=O)O)nc2ccccc2s1 C1(CN(C(C2CC(OC)C2)=O)C)C2CN(C(=O)CC3CCC(C)(C)O3)CC12 N1(C(C=Cc2ncc(C)[nH]2)=O)CCC2(CC1)CC2CNC(=O)C(C)N1CCCC1 N1(CC(=O)NCC23CC(NC(COC)=O)(C2)C3)CCC(C)(O)C1 c1(C(=O)NC(CC(C)C)CNC(=O)CCn2cnnn2)cnc2ccsc2c1 C1(NC(C2C(OC)CCC2)=O)CCCN(C(=O)Cc2c(O)ncnc2O)CC1 Cc1cc(F)c(C(=O)N(CC(C)NC(C23CC(C2)S(=O)(=O)C3)=O)C)c(F)c1 c1(C(=O)NC2CCN(C(c3cc(OC)ns3)=O)C2)cc(Br)cc(F)c1C C1(CC(=O)NCCCN(C(C=CCC)=O)C2CC2)CCCN1CC C(=O)(CCCCC#N)NCCCCC(=O)N1CC(CSC)C1 N1(C(C(N)=O)=O)Cc2ccccc2C(CNC(c2nc(O)[nH]c(=O)n2)=O)C1 c1(CC)nc(C(=O)N(C2CCCC2)CCNC(c2ccnn2C2CC2)=O)cs1 c1(C(N2CCCC(C(=O)NCCCOC=C)CC2)=O)c(Cl)ccc(F)c1Cl Cc1n[nH]c(=NCC(CC(C)C)NC(=O)CN2CC(=O)NC2=O)s1 C1(COC)(NC(=O)Cc2ccnn2C)CCN(C(=O)Cc2c[nH]nc2C)CC1 Cc1nc(C=CC(=O)NC2CCCC2NC(C2COC(=O)N2)=O)[nH]c1C C(CCNC(=O)CSC(F)F)(C(=O)NCC1CCOC1C)OC C(CCCSC)(C(=O)N1CCC(C)(CCN(CC)CC)C1)NC(=O)NC CC(C)CC(O)CC(=O)N1CCCC(C)(C(=O)N(C)CC2CCOC2)C1 CC(C)CCCCNC(c1c(CNC(c2cc(O)n(C)n2)=O)nnn1C)=O C1(C(N2C(C)CC2C(=O)N(C)CC2CCCC3CC23)=O)CC2CCC1CC2 Cn1cc(CN2CCC2(C)C(=O)Nc2cc(Cl)cc(Cl)c2F)c2ccccc12 n1(CC(N2C(C)CN(C(C3CC3C(F)F)=O)CCC2)=O)cnc2c(N)ncnc12 C(=O)(CCCCC(F)F)NC(CC)(CNC(C1CCC(C(N)=O)O1)=O)CC c1(CC)cnn(CC(N2CC(C(C)NC(=O)COC3COC3)C2)=O)c1 c1(C(C)NC2C(c3n(CC)ncc3)OCC2)cnccc1OCC c1(OC)cc(CCC(N2CCC(NC(c3csc4cncn34)=O)C2)=O)ccc1O C(C)(CC(=O)NC1(C)CN(C(C2(N3CCCC3)CC2)=O)C1)(C(F)(F)F)N(C)C C1(CC)CCc2sc(C(=O)NC3CCCN(C(=O)C(C)(C)CN(C)C)C3)cc2C1 C1(CC(=O)NC23CC2CN(C(C24CCCC2CCC4)=O)C3)CCS(=O)(=O)CC1 N1(C(=O)NC2CCN(Cc3n(CC)ccn3)C2)CC(=O)N(C)C(C)C1 C1(NC(C(CC2CC2)NC(c2ccc(N(C)C)cn2)=O)=O)CC2(CO)COC1C2 c1(OCC)ccc(OC(C)C(=O)NCc2cccc(NC)n2)c(C(=O)OCC)c1.OC c1(C(=O)OCc2ccccc2OCCC2CC2)noc2c1COCC2 C1(NC(c2c(C)ocn2)=O)CN(C(c2nc(CC3CC3)oc2C)=O)CC1CO C1(C(=O)NC23CCC(C2)C3)C2CN(CCN3CCC(C(F)F)C3)CC12 C1(NC(CC(=O)NCC)=O)CCN(C(c2cnn(C)c2C2CC2)=O)CC1C C(C)(C)(C(=O)N1CCC1CC(=O)NCc1ccc(SC)o1)SC C(=O)(C(C)(C)C(F)F)NCCCOCCNC(c1c(C)[nH]c(C(C)(C)C)c1)=O Cc1cc(C(N2CC(NC(C3CC3(C)C(F)F)=O)C2)=O)cc(Cl)c1Br c1(C(=O)NCCC2CC(CNC(CCSC)=O)C2)cn(-c2ccncc2)nc1C C(C)(CN=c1nc2sccc2c(NC(C)Cc2ccc(C(F)(F)F)cc2)[nH]1)SC O=C(C1CCCS(=O)(=O)N1)NCC1(CNC(C2CCS(=O)(=O)C2)=O)CC1 N1(C(CCc2c(C)ncs2)=O)CCCC2CCN(C(=O)C3=CCSC3)CC12 C1(N(C(c2cnc(CCC)s2)=O)C)CCN(C(=O)CCN2CCC(F)C2)CC1 c1(NCC(CC)OC)nc2ccccc2nc1NCc1nc2c(s1)CC(C)CC2 C(=O)(C1CCCc2scnc21)N(C)Cc1ccc(F)cc1F Cc1cc(Cl)cc(C(N2CCN(C(c3cn[nH]c3)=O)CC2CC(F)F)=O)c1N c1(C(=O)NCC(C)CO)ccc(O)c(OC(F)(F)F)c1 N1(C(C=C(C)C)=O)CC2(C(=O)NCC(C)(C)C3CCC3)CCC1CC2 C(C)(C(C)C(=O)NCC1(CF)CCOCC1)NC(C1(CC)CC1)=O Cc1[nH]c(C#N)cc1C(=O)NCC1C(C)CCCN1C(c1ccc(F)c(O)c1)=O C(=O)(CC(C)P(C)(C)=O)N1CCC(NC(Cn2c(C(C)C)ncc2)=O)C1(C)C C1(NC(C(CC)n2ccnc2)=O)CN(C(c2cc(Cl)n[nH]2)=O)CCC1O c1(C(N2CCN(C(C3C(OC)C3)=O)CC2)=O)c[nH]c2nccc-2c1C C#CCCCC(C)(c1nnnn1C1CCCCC1)NCC(CC)CCCC Cc1nc2ccccc2c(C)c1C(=O)NCCNC(C1CC(C)(O)C1)=O Cc1nn(C)c(CNC(=O)Oc2cc(F)cc(Br)c2)c1Br C1(N(C(C2C(CNC(C=CCN(C)CC)=O)CC2)=O)CC)CCCC1C n1(CC(N2CC3C(CNC(c4nccc(CC)c4)=O)(C3)C2)=O)cc([N+](=O)[O-])cn1 C1(C(=O)NC(C2N(C(c3c(CC)scc3)=O)CCCC2)C)CC2C(C1)C2(F)F CCC(CC(=O)NCC(CCNC(C1CC(O)CN1C)=O)OC)C1CC1 C=CC(C)(CCOC)C(=O)N1CCCC1CCCNC(c1coc(C)n1)=O CCCCC(CC)n1cc(C(C)N(C)COc2ccccc2Cl)nn1 Cc1nc2nccc(C(=O)NCC(C)N(C)Cc3coc(C4CC4)n3)n2n1 c1(OC)cc(C(=O)NCc2cccc(Cl)n2)c(-c2ccc(CO)nc2)cn1 C1(NC(C2CCC(NC(C(C)OCCOCC)=O)CC2)=O)CCC2(CCC2)CC1 C(=O)(CCCCCN(C)C)NC1C2(CC(NC(C3N(C(C)=O)CCCC3)=O)C2)C1 Cc1ccc(C(=O)NC(C)(CO)CCCl)cc1-n1cccc1 N#Cc1c(F)ccc(NC(C23CC2CN(S(=O)(=O)C(F)(F)F)C3)=O)c1F c1(C(N2CCC(C)(COC)C2)C(=O)NCCCCCC)ccc(F)c2[nH]ncc12 CCCCCCCCC(=O)N1CCCC(O)(CNCc2cccc(Cl)n2)C1 C1(CC(=O)Nc2ncc(C#C)cn2)Cc2ccccc2N1C(C)=O c1(NCC2(CC)CCCCC2)nc(=NC2CCN(CCF)C2)[nH]c2c(C)nn(C)c12 CCCC(CCCNC(c1ccc(F)s1)=O)NC(=O)C(C)(C)COC C(=O)(CCCCCNC(C1CNC(=O)C1)=O)NC(C(=O)OC)C1CCC1 C#Cc1cc(C(N2CCCC(F)(C(N3CCCC3CC(N)=O)=O)C2)=O)ccc1C Cc1nn(C)cc1CC(=O)NC1CCOC1c1nc[nH]n1 c1(-c2nc(C34CCC(=O)N3CCS4)on2)cnc2c(Br)cccn12 c1(OC)c(Cl)nc[nH]c1=NCC1(O)CN(C(=O)C(C)(C)n2cnc(C)c2)C1 N1(C(C(Cc2c(C)noc2C)C)=O)CCN(C(=O)C(C)C2CC2)CC(C)(F)C1 c1(COCC)cc(NC(=O)C=CCN(C)CC2(C)N(C(=O)CC)CC2)cc(F)n1 C1(CN(C(C(CC)F)=O)C)COCCN1C(c1ccc(OC)cc1)=O N1(C(c2c(N)nccc2)=O)CC2CCC(NC(C3CC=CCC3)=O)CC2C1 C1(C(=O)N(C2CC2)CC2CCN(C(c3c(CC)cco3)=O)CC2)CN(C)CC(C)O1 Cc1cc(O)ncc1C(N1CC(CC(=O)NCC2=CCCC2)C2(CC2)C1)=O CCCCC(CC(=O)NCCNC(=O)OC)NC(C1CC(=O)N(C)C1)=O N1(C(Cc2cc(CC)no2)=O)CCC(CNC(=O)Cc2cccnc2Cl)C12CC2 Nc1c(F)ccc(Cl)c1C(=O)NC1CCCCCC1NC(C1C2COCC12)=O C(C(C)(C)C(=O)NC1CCOC1=O)NC(C(CC=CCC)C)=O C1(N(C)Cc2c(C)nsc2)CCCC(OCc2ccccc2)C1 C1(C(N2CCC(NC(C(CC)=CCCC)=O)CC2)=O)CC2(CCC2)CO1 c1(C2(C(=O)NCC(CCNC(=O)CC3CC3(Cl)Cl)O)CCCC2)cccc(Cl)c1 CC1(C)CCCC(NCCCn2cccn2)C1 C(=O)(C(C)CC(C)(F)F)N(C1CCN(C(c2c(C)ccnc2C)=O)CC1)CC Cc1cc(CCC(=O)NC2CCN(C(=O)C=CC(=O)N(C)C)C(C)C2)cc(C)c1 c1(C(N(CC(c2nn[nH]n2)C)C2CC2)=O)cc2c(F)ccc(F)c2[nH]1 c1(C(N2CCC(O)(CNC(c3ccc(O)cc3Cl)=O)C2)=O)ccnc2ccsc12 C12(C(=O)NC3(C(NOC(C(=O)NCC)C)=O)CCC3)CSCC1C2 CCCCCCC(c1nnnn1CCC1CC1)Nc1ccc(OCC)nc1 Cc1ccc2[nH]nc(C(=O)NC3CCCC3NC(c3cc(Cl)ccc3C)=O)c2c1 C1(CNC(C2CC(OC)C2)=O)N(C(c2ccc(O)cc2)=O)CCCC1(C)C Cc1ccc(Br)cc1NC(C1COCCC1OC(C)(C)C)=O C1(NC(CCC(=O)N(C(C)C)C)=O)CN(C(c2occc2C2CC2)=O)CC1(C)C C1(CNC(c2cnn(CC)c2C)=O)CCN(C(=O)CC(C)C2CCCC2)C1(C)C C(=O)(C(C)C(O)C(C)C)NC1CC(C(=O)NC(c2ncnn2C)CC)C1 CN1CC(C)(C(=O)NCC2CCCN2C(c2cc[nH]c2C2CC2)=O)CC1=O C1(CNC(C(C)OCCC(C)C)=O)CCCC1NC(c1ccsc1C(F)F)=O C1(O)(CNC(COCCSC)=O)CCCN(C(=O)C(F)CC(C)(C)C)CC1 Cc1cc(F)c(N)cc1C(=O)N(C)CC1CCCC1NC(c1ccccc1)=O N1(C(CC(=O)OCC)=O)CCOC(C(=O)NCCOc2cccnc2)C1 CN1CC2CC1CN2C(=O)CC1CN(C(=O)CCc2ccccc2)C(C)(C)C1 c1(CC)cc(C(=O)NC2(C)CN(C(c3cccc(OC(F)F)c3)=O)C2)nn1C c1(C(=O)NC(CNC(c2ccc(OC)o2)=O)C2CC2)cccc(C(C)(C)C)c1N N1(C(C(N2CCN(C)CC2)=O)=O)CCN(c2ncco2)C2CC12.C(=O)(C(F)(F)F)N C(=O)(C#Cc1ccccc1)N1CCN(C(c2c(OC)nccn2)=O)C(CO)C1 N1(C(CCC#C)=O)CC2C(N(C)C(c3cccc(-n4cncn4)n3)=O)C2C1 N1(C(c2c(P(C)(C)=O)cccc2)=O)CCC(C(=O)O)C2CCCC12 c1(C(=O)OC)cc2c(cc1F)CCN(C(=O)NC1CCC3(CCC3)OC1)C2 N1(C(Cc2c(C)nn(C)c2)=O)CCCC(CNC(=O)C(C)Cn2ccnc2)CC1 N1(C(c2sc(C)c(O)n2)=O)CCCC(C2CC2NC(=O)CCC2=CC=C2F)C1 N1(C(CC2ON=C(CC)C2)=O)CCC(C)N(C(C2CCCN2CC)=O)CC1 c1(N2CC3CC(NC(CCC4C(C)(C)C4)=O)C3C2)ncnc2scnc12 C1(C(=O)NC(c2nccs2)C)CCC(NC(=O)Cc2cscn2)CC1 C1(C2CC2)(CNC(c2c(CC)noc2)=O)CCN(C(=O)CCOCC(C)C)C1 c1(C(N(CCCNC(=O)C(c2ccc(Cl)cc2)CO)CC)=O)cncn(C)c1=O CC(C)CC(=O)C(=O)NC1(CCC(N2CCCC2CCCO)=O)CC1 C1(OC(C)C(=O)NCC#CCNC(=O)C(O)Cc2cnn(C)c2)CCCCC1 c12cnc(cn1)CN2.C1(C(=O)Nc2nnc(-c3ccccc3)o2)CCCS1(=O)=O C1(C(N2C(C(=O)Nc3c(C(=O)OC)sc(C)c3)C=CC2)=O)CC(C)(C)CC(C)(C)C1 CC(C)(CC(=O)N1CCC1CC(=O)NC1CCC(O)C1)C1CCCO1 C1(C(=O)NC(CC(C)NC(=O)CN(CC(C)(C)C)C)C)CCc2nc(O)[nH]c2C1 C(=O)(C1=CC(C)CC1)N1C(CNC(C2(CC#C)CCCO2)=O)CC1 C(=O)(C(F)CCC(C)C)NCCCOC1CCN(C(C(C=CC)O)=O)CC1 C1(NC(C(C)CC2CCCC2)=O)CCCCC1NC(=O)Cc1ccn(C)n1 C(=O)(C=CS(C)=O)NCC(C)N(C(c1c(Cl)cnn1CC(=O)NC)=O)CC C1(CNC(CCC(=O)NCC)=O)CCN(C(C23CC(C)(C2)OC3C)=O)C12CCC2 C1(C(N2CC(C)(C)C(NC(C3(CO)CC3)=O)C2)=O)CCC2(CCCCC2)CC1 c1(COC(COC)C)cn(C(F)(F)CO)cn1 Cn1nc(C(N2CCC(NC(c3ccns3)=O)C2)=O)cc1Cl c12cc3[nH]c(cc3s1)-c1ccc(cc1)NC2=O.C(=O)(C(C)n1cccn1)OC CC(C)(CC(F)C(=O)NC1CC2CC(O)C1C2)NC(=O)C(F)C(F)(F)F CC(CC(=O)NCC(C)NC(=O)C=Cc1ccccc1Br)CC(F)(F)F S(=O)(=O)(c1cccc(=NC(C)c2nc(COC)cs2)[nH]1)N1CCC(N(C)CC)C1 CC1CC(C)N(C(c2cncc(C3CC3)c2)=O)CCN1C(c1cnc(S)[nH]1)=O N1(C(CN(C(C(NOC)=O)=O)CC2CC2)=O)CC(C(=O)OC)CC(C)C1 c1(C(N2CCC(C(C)NC(=O)COC3CCCOC3)CC2)=O)cc(O)nc(O)n1 Cc1c(C(=O)NCCNC(=O)C(c2cccc(Br)n2)C)ncn1C CCS(=O)(=O)c1ccc(Cl)c(C(=O)NC2C3CCC2CN(CC(N)=O)C3)c1Cl N1(C(c2sc(=O)n(Cc3ccccc3)c2N)=O)CCC12CCS(=O)(=O)C2 N1(C(c2cc(CNC(C3(CC)COC3)=O)nn2C)=O)CC(F)(F)C(F)(F)C1 N1(C2(C3(C(=O)Nc4ccccc4)CC3)CCC2)CC2(CC(C(=O)NCCl)CO2)C1 O=C1CCC(C(=O)NCC2CC2CNC(=O)CN2CC3CC3C2)=NN1 C12(NC(C3N(C)CC3)=O)CCOCC1CN(C(c1cncc3nc(O)[nH]c13)=O)C2 CC1(CNC(C2CC=CC2)=O)CCC(NC(c2c[nH]nc2F)=O)CC1 c1(C(=O)NCC2CCN(C(C3(SC)CCC3)=O)C2)cc(C)c2c(c1)CCC2 N1(C(C(N2CCOCC2)C)=O)CCCCC1CCCNC(C1(C)CC1)=O C1(N(C(c2cnc(CC)o2)C(=O)NCCOCC)C)CCOCC1C C1(C)(CNC(C(CC)O)=O)CCCN(C(c2c[nH]nc2-c2ccncc2F)=O)C1 CC(=O)CCC(C)(C)C(=O)Nc1ccc(C2CCOCC2)cc1C N1(C(CCOCC#C)=O)CC(C(=O)NC(C)CC2CCCC2)CC(C)C1 c1(C(C(=O)NC(C)CN(C(=O)C(C)(C)N(S(C)(=O)=O)C)C)=O)cccc(Cl)c1 C12(CC(=O)NCC#N)CCC1CN(C(=O)CN1CCOCC1=O)C2 c1(C(N2CCC3(CN(C(C4CC(C)OCC4)=O)C3)C2)=O)cc2c(cc1Cl)NCC2 C12(CNC(CC3CC(=C)C3)=O)CC(C(=O)NCCCNC(N)=O)(CO1)C2 CS(=O)(=O)c1cccc(NC(C2(O)CCN(Cc3c(O)cccc3O)C2)=O)n1 c12ccccc1C(=O)N1CC(C1)C2.C(=O)(CC(C)C1CC1)N(C(C)C)C c1(C(N(C2CCCN(C(CSCCCC)=O)C2)CCO)=O)ccc(Cl)cc1N N1(C(C(C)OCCCC)=O)CCC2(CCN(C(=O)CC(=O)OC)C2)C1 c1(OC)ccc(OC)c([N+](=O)[O-])c1C(N1CC(N(C(=O)C2=CC(C)(C)C2)C)C1)=O c1(SC)cscc1C(=O)NCC1(CNC(C2CCCN2C)=O)CCC1 C1(C2CC2)(NC(c2c(OC)nc(C)cc2)=O)CCN(C(C2(C)CCC(=O)C2)=O)C1 N1(C(COCC=C)=O)C(CNC(C2CC2c2cncn2C)=O)CC2CCCC12 c1(C(=O)NCC2CN(C(CC3CC(=C)C3)=O)C(C)(C)C2)c(C)ccc2n[nH]cc12 c1(C(=O)NC(CC)C)ccc(C(=O)OC)cc1C#N c1(C(N2CCC(C(=O)NCCC(CCC)C)C23CC3)=O)ccc(C#N)c(C)n1 c1(C(C2CCOC2)C)cn(CC(F)CCNC(=O)C(c2ccccc2)C)nn1 C#Cc1ccc(OCCOCC)cc1.c12ccc(nc1)-c1cccc(c1)C(=O)N2 C1(C(=O)NC(CC(C)C)CNC(=O)C(C)NC(N)=O)CCOCC1(C)C C1(CN(C)C)CCC(C(N2CCC(N(CCO)C(c3cocn3)=O)C2)=O)O1 c1(COC)ccccc1C(N1CCCC1C(C)(C)CNC(=O)C=CS(C)=O)=O C1(NC(=O)Cc2nc(C3CC3)cs2)CN(C(=O)C(F)C2CCCC2)CCC1F N1(C(Cc2cc(C)no2)=O)CC=CCC1C(=O)NC1CC=CC1 N1(C(C2C(C(C)NC(CN(C(C)=O)C)=O)C2)=O)CCC2(CNC(=O)O2)C1 c1(C(=O)NCC2CCN(C(c3nnn(C(C)(C)C)n3)=O)C2)ccc2c(n1)NCC2 C1(C(N2CCN(c3nc(C)nc(Cl)c3)C(C)C2)=O)Cc2nnc(C)n2C1 C1(F)(C(=O)NCCN(C(=O)CCN(C(C2CCC2)=O)CCO)C)CCOC1 C(CCC(C)(C)NC(=O)C(F)n1ccnc1)NC(C(CSC)O)=O C=CCCCCCCC(=O)N(CC(C)O)CCNC(C1CC2CC1CC2(F)F)=O C1(C(=O)NCC(=O)OC)CCCC(OC(C)(C)C)C1 N1(C(CN(C(=O)C(C2CCOCC2)=O)C2CCC2)=O)CCCC2(CC(O)C2)C1 c1(C(=O)NC2C(NC(CCNC(=O)NC)=O)C2)ccncc1-c1ccccc1.NC C(c1cnn(C)c1)=CC(=O)NCC1(C(C)NC(C(N2CC(C)C2)C)=O)CC1 CCCCC(CCCC)CC(Cc1nc(CCOC)nn1-c1ccc(SC)cc1)CC C1(C(C)C)CN(C(c2ccnnc2)=O)CCN1C(=O)CC1CCC12CCC2 C1(NC(c2cc(CCC)on2)=O)CC2CCC1CC2NC(=O)CN1CCC(C)C1 c1(CC(=O)OC(C)C(=O)NCC2CCCC2)ccc(N)cc1I c1(OC)ccc(C2(CNC3(COCC4CCOCC4)CCSCC3)CCCC2)cc1 C1(C(N(C)CC2(NC(=O)C(CSC)CC3CC3)CC2)=O)CCC(=O)NC1 C1(C(=O)OC)CCC(C(=O)OC)N1C(=O)C(C)Cc1c(C)noc1C N1(C(CC(C)(C)C#N)=O)CCc2cc(CNC(C3CCCOC3)=O)ccc2C1 N1(CC(=O)NC2C(CNC(C3(CC)CC3)=O)C2)C(=O)c2ccccc2S1(=O)=O C1(CNC(c2c(C)[nH]cc2)=O)COCCN1C(C1CC1CN(C)C)=O c1(-n2c(C(c3nc(O)n[nH]3)C)nc(CCCOC)n2)cccc2ncccc12 n1(CC(=O)NC2CCCC(NC(C3(OC)CC3)=O)C2)nc(C)c2cccnc12 C(=O)(C1=CC2(CCOCC2)C1)N1CC(CCNC(=O)CC(C)CF)(OC)C1 CCC(CC(=O)N1CCC(N(CCO)C(C2CCCO2)=O)CC1)C(C)C c1(NC(c2cncc(OC)n2)=O)ccc(C)c(C(=O)NCCC2(CC3CC3)CC2)c1 N1(C(C=C(C)I)=O)CCC2CN(C(=O)C(C)(F)c3ccon3)CC12 Cc1nc(C(=O)NC2CCN(C(C3(C(F)F)CC(=O)C3)=O)C2)cn(C)c1=O C1(CNC(C(=Cc2ccccc2)OC)=O)CCN(C(C2(C)CC2)=O)CCC1(F)F C1(C)(C(N2CC(CN(C(=O)COc3cnn(C)c3)C)C2)=O)CC2CC2C1 Cc1c(C(N2CC3C(CNC(=O)CN4CCCC(C)C4)C3C2)=O)ccn1CCO CC(C)CCC(O)C(=O)N1CCC(O)(CN(C)C(c2cc([N+](=O)[O-])cn2C)=O)C1 C1(CC(=O)NC2CC(c3ccccc3)(CNC(C3(CO)CC3)=O)C2)CCCC1(F)F C(CC(F)F)(C(=O)OC1(CC2CC2)CC1)C(C)(C)C N#Cc1n[nH]c(=NC2CCN(C(=O)CCC3CCC(=O)N3)CC2C)s1 N1(C(c2cc(OC)no2)=O)CC2(CNC(c3nccnc3C)=O)CCC1CC2 n1(CC(=O)NCC2(COC)CCCN2C(C2CCC(O)C2)=O)nc(Cl)ccc1=O N1(C(c2c(CC)cncc2)=O)CC2CCN(C(C3CC3F)=O)C2C1 Cc1ncoc1C(=O)N(CCNC(C1C(=C)CSC1)=O)Cc1ccccc1 C1(NC(c2c(C(C)C)nns2)=O)CCCC(NC(c2cc3ccsc3s2)=O)CC1 N1(C(C(C(CC)(C)C)CC(=C)C)=O)CCC(C(=O)N(C)C)=C(F)C1 c1(C(N(CC(C)NC(c2cc(C)sn2)=O)CC)=O)csc2cccnc12 Cc1nn(C)cc1C(C)C(N1CCC2C(NC(=O)CCCn3ccnn3)C12)=O C#Cc1cc(C(=O)NC2CN(C(c3cc(COC)on3)=O)CC2C)cc(Br)c1 c1(C(N2CC(C=C)C(NC(=O)C(C)NC(N)=O)C2)=O)cc2c(F)cc(Cl)cc2[nH]1 N1(C(C2C3CC(F)C(C3)N2C(=O)C=CCBr)=O)CCc2cc(Br)ccc2C1 c1(C(N2C(CNC(c3n(C)cnn3)=O)COCC2)=O)cc2nc(F)ccc2o1 c1(C(=O)NCC2CN(C(c3c(C#C)cn(C)n3)=O)CC2C)cc2cc[nH]c2cn1 c1(C(N2CCCC(N(C(C3C(C#C)C3)=O)CC)C2)=O)ccc2nn[nH]c2n1 C(=O)(C(F)(F)C=Cc1ccccc1)NCCC(C)NC(=O)C(C)OCC(F)(F)F CC(F)(F)C(C)(C)CC(=O)NC1CCCC1NC(c1cccc(C2CC2)c1Cl)=O C1(C)(C(N(CC(C(=O)N2CC(C(C)OC)C2)C)C)=O)CCCN1C C1(NC(C(C=CC)O)=O)CC2CC1CN(C(c1cncnc1C(C)C)=O)C2 c1(C(N2CC(NC(C3C(C)=C3)=O)C(C)C2)=O)cc(C#N)ccc1O C1(NC(C2(C(C)C)CCN(C(=O)C=Cc3cccnc3)C2)=O)CCCC(C)(C)C1 c1(OC)cc(C(=O)Nc2cccc(C(N3CCCC(F)C3)=O)c2)ccc1O c1(C(=O)NC(CNC(CCOCC)=O)CCOC)nc(OC)ccc1Cl N1(C(C(C2CCOC2)OC)=O)CC(C)N(C(=O)C(F)C(C)C)CC1C C(=O)(C(=O)C(C)(C)C)NC1CC(C(=O)NC(COC)C)C1 C1(N(C(c2cccc(CC)n2)=O)C)CC2CCC(C1)N2C(=O)C(F)=C(C)C1CC1 C1(C2CN(C(c3ncc(F)cc3F)=O)C2)(NC(c2occc2F)=O)CC1 Cc1ccc(Cl)cc1C(N1CCC(CCN(C(=O)C#CC(=O)N(C)C)C)CC1)=O c1(OC)nc(Cl)ccc1C(N1CCC(N(C(=O)CN2CCNC(=O)C2)CC)C1)=O C1(CC(=O)NC2(CCNC(C(C)N3CCC3)=O)CCC2)CCCC1(F)F c1(CNC(CCC(C)NC(CC2(NC(C)=O)CC2)=O)=O)c(O)cccc1F N1(C(C(C)NC(=O)C=C2CCC2)=O)CCN(C(C)(C)C)CC1 C(C(F)C(=O)N1CCCC1CN(C1CN(C(C2(O)CC2)=O)C1)C)N(CC)CC Cc1nc(C(N2CC(NC(C3(Cl)CC3(F)F)=O)C(CC(C)(C)C)C2)=O)nn1C CCC(C)(C)C(C)CC(=O)NC1C(C)(C)C(NC(=O)Cn2nnnc2C)C1(C)C c1(C(N2CC(NC(c3cc(C)[nH]n3)=O)C(C)C2)=O)c(C(C)C)nn(C)c1Cl C1(CNC(C(C)CN(C)C)=O)CCCCCN1C(c1cc(=O)c(Br)c[nH]1)=O C1(NC(c2nc(C(C)OC)sc2)=O)CC2CC1CN(C(=O)CCCCCSC)C2 N1(C(c2ncn(CC)n2)=O)CCC(C)C(CNC(c2cc(Cl)c[nH]2)=O)C1 C=CCC(CC(C)C)C(=O)NCCC1(NC(=O)CCc2ccc(C)s2)CC1 c1(N2C3CN(C(COc4cccc(OC)c4)=O)CC32)ccnc(S(C)(=O)=O)n1 N1(C(C2C(c3c(C)nn(C)c3)OCC2)=O)CCCCC(n2cc(CO)nn2)C1 C1(NC(c2c(CC)cncc2)=O)CCN(C(=O)C=CCN(C)C(C)=O)CC1O C1(CC(C)NC(C(C)=CC)=O)CC2CCC(C1)N2C(C1CC(C)CC(C)C1)=O CCC(CCOC)C(=O)N1CCC1CNC(c1cccnc1N)=O Cc1cn(C)cc1NC(=O)NCCC1CCCN1S(C)(=O)=O C12(C(N(CCNC(c3cnn(C(C)C)c3Cl)=O)C)=O)CCCN1CCC2 N1(C(N2CC(OCCOCC)C2)=O)CCC(C)CC1.Cc1n[nH]cc1C=O C1(CNC(c2ccc(SCC)cc2)=O)CN(C(=O)C(C)NC(C)=O)CC12CCC2 C12(NC(=O)CC3CSCCS3)CCCN(C(c3nc(Cl)cs3)=O)CC1C2 N1(C(c2c(N)ccc(C)c2)=O)CC2CCC1C(NC(c1nc(Cl)c(Cl)s1)=O)C2 c1(C(=O)NCC(C(C)C(C)C)NC(C=CCCC)=O)oc2ccc(C)cc2c1C c1(N(CCN(C(=O)CCc2ccn(C)n2)C)C)ccc([N+](=O)[O-])cc1Cl C1(NC(c2c[nH]cc2-c2ccccc2)=O)CCC(NC(C2OCCO2)=O)C1 N1(C(C(CCOCC)NC(c2ccc(C)nn2)=O)=O)C2CCC1CC1(CC1)C2 N1(C(CSCCC(C)C)=O)CCN(C(=O)CCc2ccc(Cl)c(F)c2)CC1C CC(C)C(O)CC(=O)NC(Cc1cnc[nH]1)C(=O)N(C1CCCC(O)C1)C C(=O)(C(C)(C)C(C)(C)O)N1CC2C(C(=O)NC(C(CC)C)CN(C)C)(C2)C1 C(=O)(C(O)C(CCC)NC(=O)C=CC=CCC)NC1(C#C)CCCCC1 C(CCCC(=O)NCC(C)C(C)O)n1cc(CN(C(C)C)CCO)nn1 c1(C(=O)NCC2N(C(Cc3onc(C)n3)=O)C3C(C2)C3)cc(Cl)c(Br)c(Cl)c1 C(c1ccc(CO)cc1)=CC(=O)NCC(CCNC(C(C)SCC(C)C)=O)(C)C C(CC(C)(C)CNC(=O)CC(C(F)F)c1ccccc1F)(OC)OC C(CN=C(NCC(C)(C)C(C)(C)O)NCC1CNCC2(C1)CC2)C(C)C.CO C(=O)(CCP(C)(C)=O)NC(C)C(=O)NCc1cnc(C2CC2)nc1 C(=O)(C1=COCC1)NC(C)C.c12ccc(cc1)SC(CC)CNC(=O)C(=O)N2 c1(C2C(C(=O)NCC(CNC(CCc3c(C)ncs3)=O)F)C2)ccc(F)cc1 C1(C(=O)NCCC(C)NC(C2(C(C)(C)OC)CC2)=O)CCCCC1C(F)(F)F c1(NC(C2CC(NC(C(C(=O)OC)C)=O)C2)=O)c(C#N)ccc(Br)c1F C1(C(N2C(C(=O)NCCCCCC=C)CSC2)=O)CCOCC1(C)C c1(C(C)NC(C2CC2NCc2ccnn2C)=O)ccccc1C(F)(F)F N1(C(c2c(Cl)cc(C)s2)=O)CCCN(C(C2CC2C2CC2)=O)CC1 c1(C(C(=O)NCC2CCC2NC(=O)CCF)=O)ccc(F)c(F)c1 N1(C(COCCCC#C)=O)CCC(C)C(NC(=O)C(C)CC=CCC)C1C N1(C(CC(CC)CC)=O)CC2(NC(C3CN=C4N=CNN4C3)=O)CCCC2(F)C1 Cc1cncc2cc(C(=O)NC(C)C(CO)NC(c3ccsc3Cl)=O)sc12 c1(N2CC3C(NS(CC(=O)OCC)(=O)=O)(CC3)C2)ncnc2cccc(F)c12 C1(C(=O)OCC)CCC2(CN(Cc3ncc(OC)cn3)C2)O1.C1(NCC)CCOCC1 c1(CC(=O)NCC2CCCCN2C(C2CCCC2F)=O)cccnc1O CC1(CC(=O)NC2CCCC2NC(c2ccn(CC3CC3)n2)=O)CCCO1 c1(OC)cc(C(=O)NC2CC(NC(=O)C(C)CC(F)F)C2)cc(F)n1 c1(C(=O)NC2CCN(C(C=NOC)=O)C23CC3)cc2ccccc2nc1C c1(CC)nc(CC(=O)NCc2cn(CCOC(C)C(=O)OC)nn2)cs1 N1(C(c2cc(C(=O)NC(=O)C3CC3)on2)=O)C2CCC1C(NC(C1CC1F)=O)C2 C1(NC(CCOCCCNC(C(C2CCC2)OCC)=O)=O)CC2CCC1O2 c1(C(N(C2CCN(C(COCc3onc(C)n3)=O)C2)C)=O)cccc(O)c1Cl C(=O)(C(C)CC(C)(F)F)N1CC(CNC(c2ccc(C)n2C)=O)OCC1 CC1(NC(c2ccco2)=O)CCN(C(=O)COC2CCCCC2)C1 c1(C(=O)Nc2cc(NC(C3CCNC3)=O)cc(Br)c2)cccc(O)c1[N+](=O)[O-] Cc1cccc(C)c1C(=O)NC1(C)CCCN(C(=O)C(C)CSC(F)(F)F)C1 C1(NC(Cc2cccc(C)c2)=O)C2CC1N(C(C1CCS(=O)(=O)C1)=O)C2C C(=O)(C(CC)CCOC)NC1C(C(=O)NCC(C=C)O)C2CCC1C2 CC1CC(NC(c2csc(C#N)c2)=O)CCN1C(c1cc(Cl)cc(Cl)n1)=O c1(OC)ccc(CC(C)(C)NC(c2ccc(C(F)(F)F)cc2)C)cc1 C1(C(=O)NCC2(O)CN(C(C=Cc3c(C)cncc3)=O)C2)CC2(COC(=O)N2)C1 N1(C(c2[nH]cc(C#N)c2)=O)CCC(F)CC1C(=O)NOCC=CCl C(=O)(CCCC(=O)N1CCCN(C(=O)C(F)n2ccnc2)CC1)NCCC c1(C(N2C(C#N)CN(Cc3ccc(Cl)nc3)CC2)=O)cccc2cc(O)ccc12 N1(C(=O)C=Cc2ccoc2)CCC(O)(CNC(C2(F)CCC2)=O)CC1 c1(C(=O)NC2CCC(NC(c3ccc(-n4cncn4)cc3)=O)C2)cncc(F)c1 N1(C(COC)=O)CC2CC(C1)CN(C(=O)CC1CCC(=O)C1)C2 c1(C(N2C(C)CCC(NC(=O)CO)C2)=O)ccc2cc(Br)ccc2c1 C(CC(=O)NC(C1CCCC1)CNC(=O)CCOC1COC1)=C(C)C N1(C(C2CCC(N(CC(C)C)C3CC3)CC2)=O)CCC12CCC(O)CC2 N1(C(c2c[nH]cc2C2CC2)=O)CC2CC1CN2C(C1CC2CCC2C1)=O N1(C(C(C)n2ccnc2)=O)CC(NC(c2ccc(C(F)F)cc2F)=O)C2CC2C1 C1(C(=O)NC(COC)C)CC(F)CN1C(c1ccc(C(F)(F)F)cn1)=O CCC(C(=O)OC)C(=O)NCCN(C(=O)C(CC(C)C)NC(N)=O)C1CC1 CC(C)C(CC(=O)NCC1=NOCC1)NC(C1CCO1)=O C12(c3onc(C(=O)OCc4cncc(C)n4)n3)CC(C)(C1)OC2(C)C c1(C(C)C)cc(=NC(CNC(=O)CCC2CCOCC2)C(C)C)[nH]c(Cl)n1 c1(C(=O)NCC2N(CC)CCC2)cc(NC(c2cc(O)n[nH]2)=O)ncn1 c1(C(C(=O)NC(C)COC)NC(CN(CCC)C)=O)cccnc1 C1(C(=O)NCCc2c(C)cccn2)CN(C)CCN1C(C1CCCO1)=O C1(CC)CN(C(c2cc(C)ccc2O)=O)CCN1C(=O)C1=C(Cl)CC1 c1(C(=O)NCC2N(C(Cc3c(C)nc[nH]3)=O)CCOC2)coc2c(F)cccc12 C(=O)(C(CC(F)F)N(C)C(C1CCN(C)C1CC)=O)NC(c1ccn(C)n1)CC C1(OC)CN(C(=O)C(C)(C)C)CC1c1cn(Cc2cn(CCCF)nn2)nn1 N1(C(C)=O)CCOC(C(N2CCC(N(C)C(c3nnn(C)c3N)=O)CC2)=O)C1 C(=O)(C(C)(C)CC(F)F)NCC(CN(C(Cc1c(C)nn(C)c1Cl)=O)C)O c1(C(N2CC(C(=O)NC(C3CCCC3)CC)C2)=O)ccc(OC)nc1Br N1(C(CC(C)O)=O)CC2CCCN(C(=O)CC3(C(F)(F)F)CC3)C2C1 c1(OCC2CCC(c3n(CCOCC)nnn3)(N(C)C)C2)cccc(Cl)c1Cl c1(NCC2CCCN(C(CC(c3c(C)n[nH]c3C)C)=O)C2)ncnc2sccc12 c12cc(ccn1)C(=O)NC2.C(C)(CC(C)CC)N(C(c1c(CC)noc1)=O)C c1(C(N2CCCC(CNC(Cc3scc(C)c3)=O)C2)=O)nnn2c1C(=O)NCC2 [N-]=[N+]=NC1CC2CCC1(NC(c1ccc(OC(F)F)cc1)=O)C2 c1(C(=O)NCCC(C)N(C(=O)C(O)Cc2ccccc2)C)ccc(C(C)(C)C)s1 c1(CCN(C2(CCC)CCC2)C(=O)C(O)C2CCC2)nc(C)oc1C CC(CCC(C)(C)C)C(=O)NC1COCC1C(N1CCN(C)CC1)=O CCCCC(C)C(=O)NCC1(OC)CN(C(C2(C)CCC23CCC3)=O)C1 C#CCCC(C(=O)NCCC1CCC(C)O1)NC(=O)CCc1cccn1C C(=O)(C(C)(C)CC1CC1)NCCC(C)NC(=O)CC1CCC(=O)O1 C1(C(N2C(CNC(Cn3nnc(C)n3)=O)CCC2)=O)CCc2nc(O)[nH]c2C1 CCCCC(O)CC(=O)N(C1CN(C(=O)Cc2ccnc(Cl)c2F)CC12CC2)C n1(CC)cnc2nc(=NCC3COCO3)[nH]c(NCc3ccc(OC)c(C)n3)c12 C1(C(=O)OC)CC2CC1CC2NC(=O)CC1OC2CCC1C2 N1(C(C(CC(CC)C)NC(c2cccc(F)c2)=O)=O)CCC2CN(C)CC2C1 C1(NC(C2(OC)CC2)=O)CN(C(C2CCOC2c2nccn2C)=O)CCC1CO CC1(C)CC(C(=O)NC2(C)CC2(C)C)N(C(C2CC3(CSC3)C2)=O)C1 C(C)(C(C)C(=O)NC1CCCC1F)NC(c1c(C(C)C)nco1)=O C(=O)(C(O)CC[S+](C)C)NC(C)C(c1ccccc1)NC(=O)C1=CCSC1 Cc1cc(C)c(C(N2CCCC3CC23)=O)c(C)c1 C(=O)(CCN=[N+]=[N-])N1C(CCC(=O)NC(N2C(=O)CCC2=O)(C)C)CCC1 c1(CC(=O)NC23CC(NC(C=C(COC)C)=O)(C2)C3)cn(C)nc1C c1(C(N2C(C)CC(CNC(c3cccc(CO)c3)=O)C2)=O)ccnc2[nH]cnc12 N1(C(C2CC(C)C2)=O)CC2CCCC2(CNC(c2ccnnc2)=O)C1 C(N=c1[nH]c(=NC(C)c2n[nH]cc2C(C)(C)C)[nH]c2c1COC2)C1CC(OC)C1 N1(C(C(C)n2ccnc2)=O)CC2CCC1CN2C(c1ccc(C#N)nc1O)=O C1(NC(C2CCN(C(c3c(C)nc(O)s3)=O)C2)=O)CCn2ccnc2C1 c1(NC(=O)NC2(Cc3c(C)ncs3)CC2)nc2c(s1)CC(c1ccccc1)CC2 C1(CCNC(COC2(C)CN(C(c3c(C)occ3)=O)C2)=O)CCCC1(C)C Cc1c(C(=O)NC2CCC(CNC(C34CC(CO3)C4)=O)C2)ncn1C C1(NC(C2C(NC(c3cn(CC=C)nc3)=O)CC2)=O)CCC(=O)NC1C CC(C)(Cc1cccc(Cl)c1)C(=O)NCCC1CC(NC(C2CC2CF)=O)C1 N1(C(C(C)n2cc(CO)nn2)=O)CCCC(C)(CNC(=O)CCN2CCCCC2)C1 C(CN=C(NCC1CCC(c2ccccc2)O1)NC1CC1)c1cc(C)n(C)n1 C1(NC(C2(COCC)CC2)=O)CC(C)CN(C(=O)CC2C=CS(=O)(=O)C2)C1 CC(C)(C)C(CNC(C1CC1(C)Br)=O)NC(CC1(CC(=O)NS(C)(=O)=O)CC1)=O c1(-c2nc(C3N(C(c4onc(C)c4Br)C)CCC3)on2)cccc(O)c1 C1(C(N2CC(CCNC(C(n3ncc(C)c3)C)=O)C2)=O)CCC(=O)N1C1CC1 C1(C(=O)NC(CNC(c2c(CC)cccn2)=O)(C)C)CC2CC(=O)C1O2 Cc1ccc2c(C(N3CCN(C(=O)CC4CCN(C)CC4)C(C)C3)=O)n[nH]c2c1 N1(C(CCc2cc(C)on2)=O)CCN(C(c2cnc(S)[nH]2)=O)C(C)C1C C1(CNC(C2(C)CC2C(F)(F)F)=O)C2CC1N(C(C1(CO)CCCO1)=O)C2 C=C(C)CCCC(=O)N(CCNC(=O)C(n1cc(Br)cn1)C)C(C)C C1(NC(C(c2ccc(Cl)cc2)C)=O)CCN(C(=O)CCc2ccon2)C(C)C1 c1(C(=O)NCC(CC(C)C)NC(C2CC2(C)C(F)(F)F)=O)cn2ccnc2s1 C1(NC(C2(CCCC)CC2)=O)CN(C(=O)CC2C(=O)ON=C2C)CC1CC1CC1 Cc1sc(S(N)(=O)=O)cc1C(=O)NC1(C)CN(C(=O)C(c2cncn2C)O)C1 N(C1CCCc2cc(CNC(=O)C3CC3)ccc21)C(C(C(C)C)n1ccnc1)=O C(=O)(C1c2ccccc2C(=O)N1C)N1CCC(F)(CNC(C(CCOC)(C)C)=O)C1 C12=CC(=NC(=O)NCCN1C(=O)C=CCF)NN2C.CC(O)COC(C)(C)C C1(C(=O)NCC(CN(C(=O)Cc2cnc[nH]2)C)O)CCC(C2CCC2)CC1 N1(C(CC2C(NC(C3(C#C)CC3)=O)CCCC2)=O)CCC(C)C(CO)C1 c1(CNC(C=CC)=O)nc(C(N2CC(c3ccccn3)C2)=O)c(C)o1 CCCCCCCCS(=O)(=O)N1CCCN(C2CC2)CC1C O=C(CC(C(F)(F)F)NC(=O)CC12CCCC1C2)N(C1(C(N)=O)CCOCC1)CC N1(C(Cc2n[nH]c(=N)s2)=O)CCN(CCNC(C2CCC(C(N)=O)O2)=O)CC1 c1(C(CC(=O)OC)NC(C2CC2C(=O)Nc2ccccc2O)=O)ccc(Br)cc1 c1(NC(C2CCC2(F)F)=O)ccc(N2CCCC2=O)cc1 c1(C(N(C2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)CC)=O)ccn(C(C)(C)C)c1 C1(NC(C2C3CN(C(C(C)c4ccco4)=O)C2C3)=O)CC2(CCC2)C1O C1(C(=O)NCCCOCCN(C)C(C2(CCO)CC2)=O)C2Cc3ccccc3C12 C(=O)(CCCC(=O)N1CCCCC1C(=O)NC1(c2nn[nH]n2)CC1)OCC c1(C(N2CC(C(=O)Nc3cccc(C(=O)NC)n3)SCC2)=O)cc(F)cc(I)c1 N1(C(C(Br)=C(C)C)=O)CCCC1CNC(c1n[nH]cc1C)=O N1(C(C2CCC(C)(C)CO2)=O)CCCC(C2CN(C(c3ccc[nH]3)=O)C2)C1 N1(C(CC=C)=O)CCOC(C)(CNC(c2cccc(CC)c2C)=O)C1 N1(C(C(C=C=C)C)=O)CC2(NC(c3ccc(S(N)(=O)=O)nc3)=O)CCCC2(F)C1 C(N=c1[nH]c(N2CCC(CC(F)F)C2)nc2cccc(F)c12)c1n(CC)nnn1 O=C(O)C1=CC2(CN(CC(O)Cn3cnc4c3CCCC4)C2)OC1 N1(C(c2nc(COC)sc2)=O)CCC(C)C(CNC(=O)C(C)(C)c2ccns2)C1 C1(C(=O)NC2CCN(C(C3(SC)CCC3)=O)CC2CO)C2CC3CC(C2)CC1C3 Cn1nnc2c(NC3CC(CNC(=O)CC4(C)CC4)C3)ncnc12 C1(C(=O)Nc2c(C)cncn2)CC12CCN(C(=O)Cc1c(F)cccc1Cl)CC2 c12cc([N+](=O)[O-])cnc1NC2=O.C1(C(N)=O)CC2COCC2N1C(=O)COCCO C1(NC(C2C(CC)C2)=O)CCC(F)(CNC(=O)CN(C)Cc2ccccc2)C1 CCS(=O)(=O)CC(=O)N1CCC(C(=O)NC(C)(C)C(F)F)O1 Cc1cc(Br)c2cc(C(=O)NC3(C#N)CC4CCCC34)[nH]c2c1 C1(NC(CCCOC(C)C)=O)CCCCC1CNC(c1ccc(C(C)O)cc1)=O C1(NC(c2c(CC)cno2)=O)CCC2(CC1)CC2NC(C1CC(=O)N(C2CC2)C1)=O C1(C(N2CC(NC(CCc3ccc(OCC)cc3)=O)C2)=O)C(C)(C)OC1(C)C N1(C(=O)NCCc2csc(CC3CC3)n2)CCCC(F)(c2ccccc2)C1 c1(-c2c(F)ncc(OCC)c2)cc(C(N2CCCC(CO)C2)=O)cc2cc[nH]c12 C1(CCC(=O)NC(CC=C)C2CC2)CCCN(C(=O)C2=COCC2)C1 c1(OC)cc(C(=O)N(CCCNC(=O)CC2CCCC2)CC)ccc1S(N)(=O)=O N(C1CCCc2ccoc21)C(C1CCC(CNC(C(C(=O)OC)(C)C)=O)CC1)=O CC(CN(C)C)CC(=O)NCCCCNC(c1cnn(C)c1C1CC1)=O C(C(CC(F)(F)F)NC(c1cccc(C2CCOC2)c1)=O)NC(CNC(N)=O)=O CCC(C)(C(=O)NC1CCCC1NC(C1CC(F)(CO)C1)=O)OC C1(NC(C2(F)CN(C(C(C)N3CCCC3)=O)C2)=O)CCN2CCCC2C1 CC(C)C(C#N)C(=O)NC1CCCC(NC(c2cc(C#N)c[nH]2)=O)C1 CC1(C)CCC12CCN(c1cc(N3CCC(OCc4ccccc4)C3)ncn1)CC2 C(CCCCCC=C)N(C(C=CCC)=O)C.C(=O)(CCS(C)=O)N c1(NC(C(C)(C)NC(c2ccc(N(C)C)cc2)=O)=O)ccccc1N=[N+]=[N-] N1(C(c2c(OC)c[nH]n2)=O)CCCCC(NC(c2csc(C)c2)=O)C1 C1(C(C)NC(C=C(C)C(C)(C)C)=O)CCCCN1C(=O)COc1ccccc1F C(CCC(=O)NC1CC(CCNC(C2(c3ccccn3)CC2)=O)C1)=CCCC C(=O)(C(O)CC(C)(C)C)N1CCC(C)CC1C(=O)NCCC(C)N1CCC1 Cn1c(C(N2CCCC(NC(=O)CCOCC3CC3)CC2)=O)cccc1=O CCC(CC)C(=O)NCC(=O)NC(C)CNC(=O)CCc1cnc(C)s1 c1(OC)cnc(C(=O)N(CCCCN(C)C(c2cnn(C)c2)=O)C)c(F)c1 C1(NC(C)(C)C)CCC2CC1CO2.C12(CCOCC1)C(C)N2.Cc1cnc(NC(=O)O)s1 C1(C(=O)NC(C2N(C(C(=O)NC(C)=O)=O)CCCC2)C)CC2CCC1O2 CCC(C(=O)NCC1CC(C)N(C(c2cc(N)cc(O)c2)=O)C1)C(F)(F)F C(CCN=C(NCCN1CCOCC1(C)C)N1CCS(=O)C(C)(C)C1)OC N1(C(c2ncccc2Cl)=O)CCC(C2CCCN(C(C3CC3[N+](=O)[O-])=O)C2)C1 c1(C(N(CC(N2CC(C#C)C2)=O)C2CCC2)=O)sc(C)cc1C C(CC(C(=O)N1CC(Cc2ccoc2)C1)NC(=O)CC(CC)C1CC1)OCC N1(C(Cc2ccc(C)cc2)=O)C2CCC(C2)C1CC(=O)NCC1C2CCCCC12 N1(C(=O)NC(c2ccc(F)cc2F)c2ccc(Br)cc2)CC2(CNCCO2)C1 c1(C(=O)Nc2c(-c3c(C)ccc(OCC)c3)csc2)cc2cc(F)c(F)cc2[nH]1 C1(NC(C(Cc2cnc[nH]2)NC(c2csc(Br)n2)=O)=O)CC2C(O)C(O)CC12 C1(N(C(=O)C=CC2(C)COC2)C)CCCN(C(c2cc(Cl)cn2C)=O)C1 N1(C(c2ncn(CC)n2)=O)CC2(CCCC2)C1C(=O)NC1CCC(O)CC1 c1(C(=O)NC(Cn2cc(CNC(C(CC)C)=O)nn2)C)cc(OC)cc(F)c1 C1(C)(C(=O)NCC2N(C(C(C)Oc3ccccn3)=O)CC2)CCCC(F)(F)C1 c1(C(CC)C(=O)NC(CNC(=O)Cn2cc[n+](C)c2)C(C)C)ccc(F)cc1 Cc1c(C(=O)N(CC(C)N(C)C(c2nocc2C2CC2)=O)C)nn(C)c1N C12(NC(=O)C3=CCC3)CCCC1N(C(c1occ3c1CCOC3)=O)CCC2 c1(CC(CN(CC(C)Cc2ccccc2)C)O)cccc2ccccc12 N1(C(C(C=C)(C)CC)=O)CC2(CCN(C(c3cncc(CC)c3)=O)C2)C1 c12nocc1NC(=O)CCN(C)CC(=O)NC2C.C1(SC(C)CO)CCC1 Cc1ccc(C(=O)N(CCCN(C(=O)CN(C2CCSC2)C)C)C)cn1 c1(C(=O)NC(CN(C(c2ccc(COC)o2)=O)CC)C)c(N)ccc(F)c1F C1(C(N(CCCNC(=O)C(O)C#N)CC)=O)CC2(C1)CC21CCC1 c1(CN=c2[nH]nc(C(C)(C)C)s2)cn2cc(F)ccc2n1 C(=O)(C(C(C)Cc1ccccc1)N1CCC(N(C)C)C(C)CC1)NC(CC)(C)C N1(C(COC)=O)CC2(NC(c3nccc4nn[nH]c34)=O)CCCC2(F)C1 C=C(C)c1cccc(NC(=O)CCOC2CN(C(=O)C=CC3CCOC3)C2)c1 O=C1CCC(C(=O)N2CCCC(O)(CNC(C3CC(C(F)F)C3)=O)C2)=NN1 N1(CC(C)C)CCN(C(=O)COC(C(c2ccccc2)C(N)=O)=O)CC1=O c1(C(=O)NC23CCN(C(c4ccnnc4O)=O)CC2C3)cc2c(Cl)ccnc2s1 N1(C(C)=O)CCC2CN(C(=O)N(C(C34CCC(CC3O)C4)=O)CCO)CC2C1 c1(CCC(=O)N(C2CCN(C(CC3CC(=C)C3)=O)C2)C)c(C)nc(SC)nc1O O=C1CC2(CCN(C(C3CCC3CNC(c3cc[nH]c3)=O)=O)C2)CN1 C1(O)(C(N2CCC(C(C)(C)CNC(=O)CCC3CCC3)C2)=O)CCCCC1 c12onc(C)c1C(=O)N1CCC(C1)N(C)C2=O.c1(NC2(CC)CC2)ccccc1 C1(NC(c2n(CC)nc(C)c2)=O)CC2CN(C(=O)C3=CCSC3)CCN2C1=O CC(C)C(C(C)NC(=O)CCc1ccccc1F)NC(c1ccnn1CCF)=O C1(CC(=O)OC)CCOCCN1c1c(OC)ccc(C(COC)O)c1 CCC(COC)C(=O)N1C(C(=O)NC2(C(=O)OC)CCCCC2)CC2CC12 Cc1n[nH]cc1CCNC(C1C(CCNC(=O)CC2(C)CCOC2)C1)=O c1(C(c2n(CC)nnn2)NCCCc2ncc(C)s2)ccc(F)c(C(F)(F)F)c1 C1(C(=O)NC2(COC)CN(C(=O)CSC)C2)CCc2nc(C(F)(F)F)cn2C1 Cc1ccc(NC(C2CC2C(=O)NCc2cccc(CO)c2)=O)c(F)c1 N1(C(C2(NC(C)=O)CC2)=O)CCCC(C2CCN(c3nnc(C(C)(C)C)o3)C2)C1 C(=O)(C(C)CC(F)(F)F)NCC1CN(C(c2cc(C)nn2C2CC2)=O)CC1C C(CCCCN=C(NCc1cncn1C)N1CCCCC(C)(F)C1)SC C(=O)(CCCCC(=O)NCC(C)CNC(c1ccc(C)c(F)c1)=O)NC C12(OC)CC(C(N3CCCC3(C)CNC(c3cc(C)[nH]n3)=O)=O)C(C1)C2 N1(C(C=CCN(C)CC)=O)CC(CNC(=O)C(C)(C)c2cccs2)C2(CCC2)C1 c1(N2C(C)C(NC(=O)CCn3cnnn3)CC2)ccc([N+](=O)[O-])cc1Br C1(C(=O)NC(CN(C(=O)C(F)=C2CCCC2)C)(C)C)CCCC2(CCCCC2)C1 c1(C(=O)NCC2CC3(CN(C(C4COC(=O)O4)=O)C3)C2)cc2sc(Cl)cc2s1 C(C1=CCCN(C(=O)CCOCCCOC)C1)NC(c1c(CC=C)cccc1)=O N1(C(C=CC(=O)OC)=O)CCN(C(c2cccn2Cc2ccncc2)=O)CC1CF c1(CC)ncnc(CC)c1C(=O)NCCCN(C)C(C1C(Cl)(Cl)C12CC2)=O c1(NC(CNC(=O)C(c2cc(Br)ccc2F)=O)=O)c(F)cc(Br)cc1Cl Cc1ccc(C(c2nnnn2C2CCCC2)Nc2cccc(Cl)c2C)c(Br)c1 C1(NC(C(C)NC(N)=O)=O)CN(C(=O)C(c2cnn(CC(F)(F)F)c2)=O)CC1F c1(C(N2CC(C(=O)NC(C(CC)C)CO)C(F)C2)=O)ccc2nccn2c1 C1(NC(C(CC)NC(=O)NC(C)(C)C)=O)CC12CCOCC2.C12CC1CNC2=O N1(C(C2C(C)C2)=O)CCOC2(CCN(C(C3(CC4CC4)CCC3)=O)CC2)C1 c1(C(=O)NC2(CCCNC(C(COC)C)=O)CC2)cccc2c1CC(C)(C)C2 C(=O)(C1=CC2(CCOCC2)C1)NCc1cccc(CNC(C(CCC)OC)=O)c1 CCC(C)C(O)C(C)C(=O)NC1CCN(C(=O)CCc2nnc(S)n2C)C1 c1(OCC2C(CNC(N3CCC3CO)=O)C2)ccc(C(F)(F)F)cc1 C1(NC(C(N2CCOCC2)C)=O)(CNC(c2ccc(F)o2)=O)CCOCC1 C(=O)(C1(O)CCCc2ccccc21)N1CCCN(C(C2(C)CC=CCC2)=O)CC1 CC1COc2c(C(N3CCCCC3c3n[nH]c(-c4ccccc4)n3)=O)cnn2C1 C1(C(=O)NC(CN(C(c2c(C)nn(C)c2Cl)=O)C)C)CCc2n[nH]c(C)c2C1 c1(C(N(C)CC2(O)CN(C(C(COC)C)=O)C2)=O)nc(OC)ccc1F c1(C(=O)NCC2(O)CCN(C(CCCCC)=O)C2)nn2c(c1Br)CCC2 N1(C(N2CCCC(C(N3CC4COCC4C3)=O)C2)=O)Cc2ccccc2C1 c1(C(C)=O)ccc(NC(c2cccc(CO)c2)=O)nc1NC(=O)C(O)C(C)(C)C CS(=O)CCC(=O)NC1CCCC1CNC(c1ccnc(Cc2ccccc2)c1)=O C12(NC(c3c(CC)csc3)=O)CCC(CNC(=O)CC3CCCCO3)(C1)OC2 c1(Cn2cc(C(CC(N)=O)NC(c3cc(Br)co3)=O)nn2)cc(Cl)cc(Cl)c1Cl C1(C(=O)NC2C(NC(CCn3c(C)ccn3)=O)CCC2)CCn2cncc2C1 N1(C(COCC=C)=O)CCN(C2CC2)CC1.C1(=O)C(OC)CN1 C1(C2CCN(C(=O)C3=CCCOC3)C2)(NC(c2cc(C3CC3)ccc2Cl)=O)CC1 N1(C(c2ccc(OC)s2)=O)CCC(NC(=O)COc2ccc(Cl)c(F)c2)C1(C)C C1(CC(=O)NC2CC(C)(NC(CCC(C)C)=O)C2)CC2CCC(C1)N2C c1(C(N2CC(COC(=O)C=CC(N3CCCC3)=O)OCC2)=O)c(Br)ncn1CCC N1(C(C2C(C)(C)NC(=O)C2)=O)CC(C2CCN(C(C3(C)CCCN3C)=O)CC2)C1 C1(CNC(C(C)(C)NS(C)(=O)=O)=O)CCCCCN1C(C12CC(O)C1C2)=O N1(C(C(C)SCC)=O)CCCN(C(=O)CCC(=O)NC(C)C)CC1c1ccccc1 N1(C(C(CC#C)C2CC2)=O)CCOCCC1C1CC1 C=CC(C)(O)C(=O)NCC1(CNC(=O)CN2CCCC2C)CCCC1 C1(C(=O)OCC)CCC(C(=O)OC2C(COC(=O)OC(C)(C)C)C2(C)C)CC1 C1(C(=O)Nc2cccc(OCCC)c2)CC12CC(C)(C)C2 C1(COC)CNCCN1C(c1ccc(-c2cccc(C(N)=O)c2)cn1)=O c1(C(N(C(C)C)CCNC(=O)C(C)S(N)(=O)=O)=O)ccc2cccc(F)c2n1 C1(CNC(c2n(CC)ncn2)=O)(NC(=O)Cc2ccn(C3CC3)n2)CC12CCC2 c12ncccc1CSCCC(=O)NC2.c1(CNC(CCC#C)=O)ccc(F)cc1 c1(C(=O)NCCOC(CNC(C2C(C#C)C2)=O)(C)C)coc2c1NC(=O)CCC2 c1(CN2C(CC(=O)NCC3(F)CCOC3)COCC2)cc(Cl)ccc1F C1(NC(c2c(C)nc(CO)s2)=O)CN(C(=O)Cc2cc[nH]c2)CC1S(C)(=O)=O c1(C(N(CCN(C(C=CC(=O)N(C)C)=O)C)C)=O)ccc2sccc2c1 c1(-c2cc(C(=O)OC)sc2C)cnn2c1CN(c1ncnn3ccc(Br)c13)CC2 N1(CC2C(=O)NCCC2)CCCCC2(CCN(C(=O)C3=CCCCO3)C2)C1 Nc1nc(C(=O)NC2CCN(C(c3ncoc3C(F)(F)F)=O)C2)cnc1Br C1(NC(=O)NC2C(CC)CN(S(C)(=O)=O)CC2)CC(C)(C)CC(C)(C)C1 C(CCCC(=O)NCC1(CNC(c2cc(C3CC3)on2)=O)CC12CCC2)OC.COC C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C2CN(C(c3c(C)cccc3C)=O)C1C2 C#CCCN=C(NCC1(C(=O)OC)COC1)NC1CCCCC1 N1(C(C2(C)CCCC2(F)F)=O)CCCCCC(NC(c2ccnn2C2CC2)=O)C1 C1(C(=O)NCCn2nccn2)CCCC(NC(C2(CO)CCCCC2)=O)CC1 N#Cc1ccc2c(C(=O)NC3C4CN(C(c5ccc[nH]5)=O)CC34)c[nH]c2c1 C1(C(=O)NCC2C(NC(c3cnc(CCC)s3)=O)C2)CCC(=O)N(CC)C1 C1(C(F)(F)F)(NC(C(C)=O)=O)CCC(F)(F)CC1.c1(N2CC2=O)ccccc1F C(=O)(N=c1cc(C)o[nH]1)c1c(NC(C(c2nccc(C)c2)(F)F)=O)cccn1 CCC(CCCC(=O)N1CCC(NC(=O)C=CCOC)C(C)C1)OC C(=O)(CCC(C)(C)C(=O)N(CC(C)NC(c1c[nH]nc1-c1cccs1)=O)C)OC Cc1cc(C)n(CC(N2CCC(N(C(C)CC#N)CC3CCCO3)CC2)C)n1 N1(C(C(C)n2ccnc2)=O)CC(C(=O)N(C)CC2(C)CCCC2)CC12CCC2 c1(C(=O)C(C2CCN(C(C3CCC3C(F)F)=O)C2)OC)ccccc1 c1(C(N2CCC(C(=O)NC3(C#C)CCOC3)C(O)C2)=O)cc2ncccc2[nH]1 Cc1ncc(N)cc1C(N1CCC(C)(C)C1CNC(=O)CC1(O)CCOC1)=O CC(C)(F)CCC(=O)NCc1nc(C(=O)NC2CCOC2C2CC2)co1 C1(CNC(C(C=C)(C)C)=O)CC2(CCN(C(=O)CN(CC)CC)C2)CO1 c1(C(N(C)CC2CCCN(C(CCNC(=O)NC)=O)C2)=O)nccc(N)c1Cl Cc1c(C(=O)NC(C)(CNC(C2(F)CCC2)=O)CO)cnn1CCO C(=O)(CC1CNc2ccccc21)N1C(C#C)CNCC1 N1(C(C(c2ccc(F)cc2F)C)=O)CCCC(N(C)C(C2(C)CCCS2)=O)CC1 C1(NC(c2c(C)c[nH]c2)=O)CN(C(c2cocc2C)=O)CC1C(F)(F)F C1(CC(C)C)(C(=O)OCCOCCCCN2CCOCC2)CCCN(C(C)=O)C1 c1(OC)cccc(CC(=O)NC2(CF)CN(C(=O)C(C)(C)C3CCCO3)C2)c1 c1(C(=O)NC(c2ccc(Cl)o2)C)ccc(OC(F)F)cn1 C1(NC(C2(n3ccnn3)CC2)=O)CCN(Cc2ccnc(CO)n2)CC1 c1(OCCCOC(COCCNC(CC2C(C)C2)=O)(C)C)c[nH]cc(Cl)c1=O N1(C(C2C(CC)CCO2)=O)CC(NC(c2cccc(F)c2OC)=O)CC(C)C1 C1(CCOCCN(C(CCC)=O)C)CC(NC(=O)C(C)NC(=O)OC(C)(C)C)C1 c1(NCCC2CN(C)C2)nc(N2CCS(=O)CC2)nc2sccc12 C1(NC(C2CCC(C)S2)=O)(CNC(c2cc(N)nc(Cl)c2)=O)CCC(C)(C)CC1 Cc1cccc(C(=O)NCCC2C(C)CCCN2C(=O)CC(C)(C)C2CC2)c1C c1(C2(NC(=O)NCCC(C)NC(C(CC)C(C)C)=O)CC2)ccc2c(c1)OCO2 CCC(COC)C(=O)NC(C(=O)NCC(C)=C(C)C)c1ccco1 CC1CC(CNC(C2CCC(F)CC2)=O)CN1C(c1ccsc1)=O C1(CC(=O)NCCCN(C)C)CCCC1 n1(CC)ncc(C(C(=O)NCC2CCOCC2)N(C)Cc2cnco2)n1 c1(C(C)C)ccc(F)cc1C(=O)NC12CC1CN(C(=O)CCc1cnoc1)C2 C(=O)(C(O)CCS(C)=O)NC1(CNC(c2cc(C(=O)OC)[nH]c2)=O)CC1 N1(C(c2n(C(CC)C)ncc2)=O)CCN(C(C2(C)CC(F)(F)C2)=O)CC(C)(F)C1 c1(CC(=O)NC2CC(OCC(=O)N(C(C#C)C)CCCC)C2)ccn(C)c1 c1(C(=O)NC(CC(F)(F)F)c2ccc(Br)cc2)ccc2c(c1F)CCC2 N1(C(=O)Cc2cc(C3CC3)on2)CCN(CCF)CC1 CN1CCN(CC(N2CCCC(N(C(=O)Cc3c[nH]nc3O)C)C2)=O)CC1 C(C)(CCCN=c1nc(N(C)CCN(C)C)c2[nH]ccc2[nH]1)SC C(=O)(C#CC(C)(C)CNC(c1cc(O)cc(F)c1)=O)NC1(C#C)CC1 c1(C(=O)Nc2ccncc2)cc(N)ccn1.C1CCCCNC(=O)CN1C c1(OC(C)C)ccc(S(=O)(=O)N2CCCN(C=O)CC2)cc1Br c1(C(=O)NCC(C)(C(C)C)NC(C(CC=CC)C)=O)ccn2ccsc12 C1(OCC)CCN(Cc2noc(-c3ccc(OCC)cc3F)n2)CC1C N1(C(CC=C)=O)CCCCC1c1cccnc1CN(C)Cc1cncn1C c1(C(=O)NCCN(C(C(C2CC(F)(F)C2)OC)=O)CC2CC2)occc1Br C1(C(=O)NCC(CC=C)NC(=O)C(=O)Nc2ncc[nH]2)C(F)(F)C12CCC2 n1(CC)ccc(C(=O)NCCCN2CCC(NC(C3CCC(O)CC3)=O)C2)c1C C1(C(=O)OC)CC2(CN(C)CCNC(C34CC(CC(F)F)(C3)C4)=O)CC1C2 Cc1cc(CC(=O)NC2(CF)CCN(C(C3OCC3(C)C)=O)C2)c(C)s1 c1(OC)cc(Cl)c(C)cc1C(=O)NC(CNC(c1cc2ccccc2s1)=O)CO O=C(C=Cc1ccc(-c2ccccc2)o1)N=c1ccn(-c2ncccc2Cl)[nH]1 C1(C(=O)N(C2CCC(NC(C3CCCC34CC4)=O)CC2)C)(COC)CCC(=O)N1 CC1(CNC(=O)CC2CC(F)(F)C2)CCCN(C(C2CC(O)C2)=O)C1 c1(C(N2CC(CC(CNC(C(CC)(C)CC)=O)(C)C)C2)=O)nc2ccccn2c1F CC1CCOCC1C(=O)NCC1(CCNC(C23CC(CO)(CO2)C3)=O)CC1 N1(C(C2(CC)CC2)=O)CC2(CCN(Cc3ccc4oc(=O)n(C)c4c3)CC2)C1 N1(C(c2cnsn2)=O)CCCOC(CCNC(C23CCCC2OCC3)=O)C1 C1(C(=O)Nc2ccc(N(C(=O)CCS(C)=O)CCOC)cc2)CCC(C)(F)CC1 c1(CCCC(=O)NC23CC(NC(c4c(OC)csc4)=O)(C2)C3)cccc(C)c1 n1(CC(=O)NCC(CN(C(CCC(CC)C)=O)C)(C)C)nnc2c1CCCC2 C1(CC(=O)NC(C(=O)OC)(C)C)CN(C(=O)C=CC2CCOC2)CCC1C C1(NC(C(C2CCC2)OC)=O)CC2(C1)CC(NC(=O)CCCc1cnn[nH]1)C2 N1(C(c2c(F)ccc(N)c2)=O)CC(C2CN(C(=O)CC3CNC(=O)O3)C2)C1 N1(C(C(C2CC2)OCC)=O)CC(NC(c2ccsc2OC)=O)C2CC2C1 c1(CC(N2CC(C(C)C)N(CC3CCCC3)CC2)=O)cc2ccncc2[nH]1 C(=O)(C1Cc2ccc(F)cc21)N1CCC(CNC(C=CC(=O)N(C)C)=O)C12CC2 C1(C(N2CC(OCCOC)C2)=O)(OC)CCN(C(c2ccc(C#N)o2)=O)CC1 c1(COC(=O)CO)ccc(Cl)c(Cl)c1.c12cccc(c1)NC2=O C#CCCCC(C)C(=O)NCc1cc(C(=O)N(CC(F)(F)Cl)C)no1 CC1(C)CCC2(CC1)CC2c1nc(CCO)nn1CC1CC(F)(F)C1 c1(N(C(=O)C(C)(C)C)CCCOC(C(COCC)C)=O)ccc2c(c1)OCCO2 c1(C(N2CCN(C(CCC=C=C)=O)CC2CCC)=O)cc2cc(C)ccc2[nH]1 C=C(C)CN=C(NCC(c1ccccc1SC)(F)F)NC1CCSC1 C1(NC(c2c(OC)n[nH]c2)=O)COC2CN(C(c3cnncc3O)=O)CC12 N1(C(c2cc(C)n(C)n2)=O)CCC(N(C)C(c2cc(Cl)cnc2O)=O)C2(CC2)C1 C1(C(N2CCC(=CCNC(c3ncc(C(F)F)s3)=O)CC2)=O)CCC2(CC1)N=N2 c1(OC)cccc(CN2CCC(O)C(C(C)(C)C(N3CCSCC3)=O)C2)c1F C1(CNC(CCCOCCOC)=O)CCCCN(C(c2cn(C(C)C)nn2)=O)C1 c1(C(=O)NCC(C(C)C)NC(=O)C(C)(C)c2cc[nH]n2)ccc2ccncc2c1 C1(NC(c2cnc(-c3ccc(C)o3)s2)=O)(CO)CCCN(C(C2CC2F)=O)C1 C1(NC(C=C(C)Cl)=O)CN(C(=O)Cc2csnc2C)C2CC12 c1(CC(=O)NCCCNC(c2cnn(C3CCOC3)n2)=O)cnn2c1CCCC2 C1(CCC)CN(C(c2c(Cl)nsc2Cl)=O)CCN1C(c1cn(C2CC2)nn1)=O N1(C(CCCSC)=O)CCC2C(NC(c3cccc(OCC(N)=O)c3)=O)CC12 c1(C(N2C(CNC(=O)C3=NOCC3)C(C3CC3)CC2)=O)cc2n(n1)CC1(CC1)C2 N1(C(CCC)=O)CCC(N(C2CCN(C(C)C)C2=O)C(=O)CNS(N)(=O)=O)CC1 c1(CCC(=O)NC2C(CNC(C(C)CN(C)C)=O)C2)ccc2c(c1)OC(F)(F)O2 N1(C(C=C(C)c2cccs2)=O)CCC(C)(C)C(NC(=O)C=C2CCC2)C1 C1(CCC=C)(C(=O)NC(C)CCC2CC2)CN(C(C2CC2CC)=O)C1 c1(C(=O)NC2CC2)nc(=NCC2CCCCN(SC(F)F)C2)cc[nH]1 N1(c2n(CCC=C)c(C3(SC)CC3)nn2)CCC(C(=O)OC(C)(C)C)(CO)CC1 c1(OC)ccccc1CC(=O)N(C)CC1CN(C(C2(O)CCOCC2)=O)C1 CC(C)CCC(F)C(=O)NCCC1CC(F)(F)CN1C(c1ccn(C)n1)=O CC1(NC(=O)C(F)CC2CCOC2)CCN(C(=O)C2=CCCC2)C1 CC1CC(NC(=O)C=Cc2cccc(Br)c2)CCN1C(=O)C(=O)NCC1CC1 C1(C(N2C(C)CN(C(=O)CCOCC3CC3)CCC2)=O)CC2(CCOCC2)CO1 c1(OC)ccc(CC(=O)NC2CC(C(N3CCCCC(C)C3)=O)C2)c(C)c1 C1(CC(=O)NCC(CC)CO)CC(O)CN1C(C1(COC)CCNC1=O)=O N1(C(C2N(C(CNC(CC)=O)=O)CCC=C2)=O)CC(=O)NCC1CC C(CCCC(CO)NC(=O)CN1CCCC1)NC(C(CCC)O)=O CC1(C(N2CCN(c3ccc(-c4nn[nH]n4)cc3)CC2)=O)CCCNC1 CC1=C(C(=O)NC2CCN(C(c3c[nH]nc3F)=O)C(C)C2)CCCO1 CC(C(=O)NCCCN(C(C1(Br)CC1)=O)C1CC1)n1ccnn1 N#Cc1cnc(NCCC2CCC(NC(c3cc4sccc4cn3)=O)C2)c(F)c1 N1(C(C(N)=O)=O)CC2CS(=O)(=O)CC2(NC(C2CC=CCO2)=O)C1 c1(NC(c2c(F)ccc(C)c2)=O)sc2c(c1C(N1CCC(C)(O)CC1)=O)CCCC2 C1(NC(CC(CC)C2CCC2)=O)CC(OC)CN(C(=O)C(C)(F)F)C1 c1(NC(C)=O)ccc(Cl)cc1NC(=O)Cn1ncc(C)cc1=O N1(C(C(C2CN(C(C3CC3(Cl)Cl)=O)C2)OC)=O)CCOCC(C)(O)C1 Cc1c(C(N2CCCC2CNC(=O)CCC2CC2C)=O)ccn1CCO N1(c2cc(OC)nc(C(C)C)n2)CCCC(C2(NC(c3cncnc3)=O)CC2)C1 c1(O)cc(Cl)c(CN2CCC(COC)C2)cc1OC.c1(CC(=O)CC)ccc(Br)nc1 N1(C(Cc2ccc(C(C)=O)cc2)=O)CCC2CN(C(c3coc(C)c3)=O)CC12 c1(C(N2CCCC(CNC(C3C(C)=C3)=O)CC2)=O)n[nH]c2c1CC(C)CC2 C1(OC)CN(C(=O)C(O)CN(C(=O)Cc2cc(C)nn2C)C2CC2)CC12CC2 N1(C(=O)C2=CCSC2)CC2(C1)CN(C(c1cnn3c1CC(F)(F)C3)=O)CCO2 c1(CNC(C2(COC)CN(C(C3CC3C(=O)OC)=O)C2)=O)cccc([N+](=O)[O-])c1 CCCCC(F)C(=O)N1CCCCCC1CNC(C12COCC1C2)=O c1(C(N2CC=CC(NC(C(C(C)C)N(C)C)=O)C2)=O)cc(N)c(Cl)c(O)n1 c1(C(=O)NCCC2CN(C(=O)Cn3nccn3)CCO2)scc2c1OCCO2 CCC(CC(=O)N1CC(CCNC(c2cc(C)no2)=O)C1)C1CC1 C1(N(C(C(c2cccs2)SC)=O)C)CN(C(=O)CCn2cc(C)cn2)CC12CC2 C(=O)(C(C)CC(=O)c1cccc(F)c1)NCC(C)OCCOC c1(C(C(=O)NC2CC(NC(=O)C=CCN3CCC3)C2)F)cccc(F)c1 C(c1cc2c(cc1Br)OCO2)=CC(N1CCC(N(CC)CC)CC1)=O CCCCC(CN=c1[nH]c(C2CC2)nc(=N)[nH]1)NC(=O)C(C)C1CC1 C1(C(=O)Nc2n(C)nc(Cl)c2)CC2CCC1N2C(=O)Cc1ccco1 c1(C(=O)NC2(CNC(CC3C(C)C3)=O)CC2)ccc2nccn2c1 Cc1ncc(N)cc1C(=O)N(C1CCCC1)CCCNC(=O)C(C)C(C)O C1(NC(C2CC3(CC(=C)C3)C2)=O)CN(C(=O)Cn2cc(Cl)cn2)C2CCCCC12 N1(C(c2nc(NC(C)=O)sc2)=O)CCC2(CCN(C(=O)CC3=NNC(=O)C3)C2)C1 C1(CC(=O)NCCCC(=O)N(C)C)CCN(C(C2CC2C2CC2)=O)C1(C)C C(C(CNC(=O)C=CC(C)(C)C)S(C)(=O)=O)NC(C1(CC=C)CC1)=O N1(C2CN(C(c3conc3C)=O)C2)CC(CC)CC1=O.N12CCC1C2=O Cc1nn(CCC(=O)NCC(C)CNC(=O)CCSCC(C)C)cc1Br N1(C(C2CCC(C(C)C)CC2)=O)CC2(NC(c3cnn[nH]3)=O)CCC1CC2 C1(NC(C=CCC2COCC(C)O2)=O)CCC12CN(C(=O)CC=CC(C)(C)C)C2 CCCCCC(O)CC(=O)NCC1COC(C)(C)CN1C(C1CC(N(C)C)C1)=O CC(C)(C)C(=O)CCC(=O)NC(CO)C(=O)NCC(c1ccncc1)O c1(C(=O)NCC2CCC(NC(C(CC#C)C)=O)C2)cc(C)ccc1NS(C)(=O)=O Cc1cc(Cl)nc(Cl)c1C(N1CCC(CC(=O)NC2CCCC(F)(F)C2)C1)=O c1(C(=O)NCCOCCNC(Cc2nc(CC)sc2)=O)ccc(O)nc1Cl N1(C(CC(COC)C)=O)CCC(C)(C)C1CNC(c1cc(O)n(CC)n1)=O c1(OC)cncc(CNC(=O)CC2CCCN2C(=O)CC2CC(SC)C2)c1 N1(C(C2C(C)CCO2)=O)CCOC(C)(CNC(C2CCC(CO)CC2)=O)C1 C1(C(C)(C)C)CCCN1C(=O)NCCSC1CCCO1 c1(C(=O)NC(CCNC(C(C=C)(C)O)=O)C)ccc2nn(C)cc2c1 N1(C(c2c(CC)cns2)=O)CC(OC)C(C(=O)NCCOC2(C)CCCC2)C1 N1(C(c2c(CC)n[nH]c2)=O)CCC2CC2(C(=O)NCC2CCCO2)CC1 C1(NC(C(=O)NCC)=O)CN(C(C2CCNC2=O)=O)C2(CCCCC2)C1 C(CCCCC(=O)N1CC2CC1CC2CO)C(NNC(C1C(N)CCCC1)=O)=O C1(OC)CCCCC1NC(=O)NCCCCCF Cn1nc(O)cc1C(N1CC(O)(CCNC(=O)CCCCc2cnn[nH]2)C1)=O C1(C(=O)NCC2(F)CN(C(CCCCCOC)=O)C2)CCC2(CCOC2)O1 N1(C(c2cccc(CC)c2C)=O)CC2CCC(C1)N(c1nccc(C)n1)C2 C1(Cc2n(CC)c(N3CCC(F)(F)C(F)C3)nn2)CCc2ncc(Br)n2C1 CC1CC2CN(C(=O)CCC3CCC3)CC2N1C(c1ccc(Br)s1)=O N1(C(C2N(C(c3c(C)n(C)nc3)=O)CC=CC2)=O)CCN2CCC1C2 C(=O)(C1=CC(O)CCC1)NC(C(C)C)CNC(c1cnc(C(C)O)s1)=O N1(C(CC2C(C)CC2)=O)CCCC12CCN(C(c1ncc3n1CCCC3)=O)CC2 c1(C(N2CCC(CCC(=O)NCC(C(C)(C)F)(C)F)C2)=O)c[nH]c2nccc-2c1 C1(CC(=O)NCCC2N(C)CCC2)COCCN1C(=O)CCC(=O)c1ccc[nH]1 N1(C(COCC)=O)CCC(C)C(CNC(=O)Cc2ccncc2Cl)C1 CCC(C)(C(=O)NCC(O)CCNC(=O)Cc1cc(C)n(C)n1)C(N)=O C(=O)(CCCCC(F)(F)F)N1CC(NC(=O)C(O)C2CCCC2)CC(F)(F)C1 c1(C(C)C)ccc(C(=O)NC2CC23CC(NC(=O)CC2CCCN(C)C2)C3)cc1 N1(C(COCCCCCC)=O)CCN(C(=O)CCc2cccnc2C)C(CC)C1 c1(C(=O)NCC2CCC(NC(CCCCSC)=O)CC2)ccc(C#N)c(Cl)c1 C(CC(C)C(=O)N1CCC(NC(=O)CN(C)C(=O)C2CC2)CC1)OC C(C#CC(=O)NC(C1(C)CC1)CO)NC(C(C)NC(=O)OC(C)(C)C)=O C(=O)(C1=CC2CCCC12)N1CCC(NC(=O)CCc2cc(F)ccc2F)(CF)C1 C(=O)(CCCCC(C)=O)N1C(C(=O)NCCC(CCC)O)CSCC1 N1(C(C(C)Oc2ccccc2)=O)C2CCC1CN(C(C1CCN1S(C)(=O)=O)=O)C2 c1(OC)ccc(OC)c(Cl)n1.C12CCN(C1)C(=O)CONC(=O)N2.C(CO)CC N1(C(CCOC)=O)CCC2(CC1)CN(C(C1CN(C)CC1(C)C)=O)CCO2 C(=O)(CCC(C)(C)F)N1CC(CNC(C(C)Sc2ccc(C)cc2)=O)C(CO)C1 C1(NC(C2C(C)CCOC2)=O)CC2CCC1CN2C(C1(C)CCC1)=O Cc1cc(C)n(-c2cc(-c3nc(C4CCC(=O)NC4)n(CCCO)n3)ccn2)n1 C1(C(=O)NCCCNC(CN(C(=O)CC(C)C)CC#C)=O)CCS(=O)(=O)C1(C)C N1(C(c2n(C(CC)C)ncc2)=O)CCC(O)(CNC(C2CCC(=O)O2)=O)CC1 C12(C(=O)NCC3CCCN(C(CCC)=O)C3)C(N)C3CC1C2C3 c1(SCC(CC)N2CCCC2)ccccc1NCc1cc(NC(=O)OCC)no1 Cc1cn(C)cc1C(=O)NCc1cccc(C(=O)NOC2CCOC2)n1 C1(NC(C(C(CC)C)C)=O)CN(C(c2ccc(O)cc2Cl)=O)C2CCCCC12 N1(C(c2ccc(C)c(C)n2)=O)CC2(CCN(C(=O)C=CC3COC(C)(C)O3)C2)C1 C1(CNC(Cc2c(CC)con2)=O)CC(OC)CN1C(=O)Cc1csnc1C c1(CNC(C(C)CSC(F)(F)F)=O)cccnc1CNC(=O)CC(C)CN(C)C N1(C(CCC(=O)NC)=O)C(C)CC2CN(C(c3nn(C)cc3C)=O)CC12 C(=O)(CCO)C1(C(=O)NCCOCCCNC(C2(CSC)CC2)=O)CC1 c1(C(=O)NCC(C)NC(=O)C2=NNC(C(F)(F)F)C2)cc(Cl)c(Cl)[nH]c1=N C12(CCN(C(=O)NCC3Cc4ccccc4O3)CCO)CC3CC(CC(C3)C1)C2 CC1(C)Cc2[nH]nc(C(=O)NC3(C)CC(NC(=O)Cn4[nH]cnc4=N)C3)c2C1 Cc1ccc(OCC(=O)NCC(C)(C)CCNC(C2(C)CCCCC2)=O)c(F)c1 N1(C(c2cccc(OC)c2)=O)CCCC(NC(=O)CCN2CCCS2(=O)=O)C1C C1(CNC(C(N2C(C)CCCC2)=O)=O)CN(C(=O)OC(C)(C)C)CC1(C)C Cc1cc(C(C)NC(=O)C(C2CCC2)NC(=O)CC2COCCO2)no1 c1(OC)cc(C(=O)NCC2COC(CNC(C3CCCCC3O)=O)C2)cc(C)n1 c1(CCOC)cncn1CCNC(=O)C(=O)OC(C1CCCC2CC12)=O C1(CN2CCC(CNC(Cc3ccc(OC)cc3)=O)C2)CCCS(=O)(=O)C1 C1(NC(c2c(CC)non2)=O)CN(C(=O)C(CO)N(C)C)CC1C c1(COC(COC(=O)NC2CC(C)(C)NC2=O)=O)cc2cccn2cn1 c1(NC(C)=O)cccc(O)c1.CCC(O)C(=O)C(C1(C(=O)OCC)CC1)=O C1(CC)C(C(=O)NCC2CCCS2)CCCN1C(=O)C(C)OC(C)=O Cc1noc(CN(C2CCC(NC(C(C)O)=O)C2)C)n1.C(CCN)O C1(C(=O)NC(C)CNC(c2c[nH]c(Br)c2)=O)CCN(C(=O)OC(C)(C)C)C1 C1(SC)CN(C(c2cccnc2N)=O)CC1NC(C1CCC(C(N)=O)CC1)=O N1(C(c2ccc(CC)o2)=O)CCC(O)(CNC(C2CSC2)=O)CC1 Cc1ccc(C#N)cc1NC(C)(CCc1ccccc1F)c1nnnn1C1CC1 c1(C(=O)NCC(CCNC(C2(C#C)CC2)=O)O)c(C(F)(F)F)cccc1CC c1(C(=O)NCCNC(C2C(C(=O)OCC)C2)=O)cc2cc(F)ccc2s1 n1(CCC=C)c(COCC)nnc1-c1ccccc1N(C)C.c12nnc(s1)SC2C N1(C(CC(=C)Br)=O)CC(C2CCN(C(C3CCCN(C)C3)=O)CC2)C1 N1(C(c2cc(CC)oc2C)=O)CCCC(CCNC(C2(CC)CCOC2)=O)CC1 C1(CNC(CCC)=O)CCC(C(N2CCN(CC3CCCO3)CC2)=O)CC1 C=C=CC(C)C(=O)N(C(c1ccccc1)CNC(c1cnn(C(F)F)c1)=O)C C12(NC(c3sc(C)c(Br)n3)=O)CCC(C1)N(C(C1CCCCO1)=O)C2 C12(CNC(c3cncc(OC)c3)=O)CCC1CCN2C(c1cc2occc2[nH]1)=O c1(OCC(=O)NCC(CNC(=O)COC2CCOC2)O)ccc(Br)cc1.C(CO)O Cc1cc(Cl)c(CNC(=O)CC2CCC(NC(=O)Nc3occc3C)C2)cc1F C1(NC(C2(CC)CC2)=O)CN(C(c2ocnc2-c2ccccc2)=O)CC1O n1(CCCOC)nc(C(=O)NC(C)CNC(c2cc(Cl)cs2)=O)ccc1=O c1(C(N2CC3C(C(=O)NCc4cnccn4)C3C2)=O)cccc([N+](=O)[O-])c1I c1(C(C)C)cc(NC(N2CCC(c3ncc(Cl)cn3)CC2)=O)cc(C(F)(F)F)c1 CC1CC(NC(=O)CCc2cccnc2)CN1C(=O)C(=O)NCC1CC1 C12(C(=O)NCCCC3N(C(CCN(S(C)(=O)=O)C)=O)CCC3)CC=CC(C1)OC2 c1(CCC)cc(C(=O)NCc2ncnn2CCF)ccn1 N1(C(C=CC=CCC)=O)CC=C(CCNC(=O)CCC(=O)N2CCOCC2)CC1 C=C(C)CC(C(=O)NC(CC(C)C)C(=O)OC)NC(=O)Cc1ccoc1C c1(C(N2CC(C(C)NC(c3c[nH]cc3Br)=O)OCC2)=O)c(F)cc(Cl)cc1F C1(n2ncc(C(N(CCC(C)NC(C(C)NC(N)=O)=O)C)=O)c2)CCS(=O)(=O)C1 N1(C(CCc2cnc(C)s2)=O)CCOC(CNC(=O)CCc2cn(C)nc2C)C1 CCCC(C(O)C(=O)NCCCCNC(=O)NC)NC(C1(C)CCN(C)C1)=O c1(N(C)C(c2nnnn2-c2ccccc2)C2C3CCCC23)nc2c(n1C)CCC2 CC1(C)C(C(N2CCCC(NC(=O)CCF)C2)=O)CC12CC(=O)C2 c1(C(N(CCN(C)Cc2nc(C)[nH]n2)C(C)C)=O)c2ccccc2nn1C N1(C(COCCCNC(C(CC)COC)=O)=O)CCC12CCC(C)CC2 C#CCC(C(=O)N1CC(CC)C1C(C)C)NC(C1CCOC1C(C)C)=O Cc1c(Cl)ccc(C(N2CCC(=CC(=O)Nc3cc(F)c(Cl)cn3)CC2)=O)c1Cl c1(OC)ccc2c(c1)CCCC2CNC(=O)NC1CCC(NS(=O)(=O)C(C)C)C1 c1(-c2c(CCC)ocn2)nc(-c2cccc(F)c2)nn1C(C)C N1(C(c2n(CC)cnn2)=O)CCN(C(C2(CN(C)C)CC2)=O)CC2CCCCC12 c1(C(=O)NC(C(N2CC(OCC#C)C2)=O)C2CCCC2)ncncc1N CC1COCCC1C(=O)NCCCOCCN(C)C(c1ncoc1C1CC1)=O N1(CC2CN(C(C3CC(Cl)(Cl)C3)=O)C2)CCN(C(C2(O)CCOC2)=O)CC1 N1(C(C(Cn2ccc(C)n2)C)=O)CC(N(C)C(c2nnc(C)s2)=O)C(O)C1 c1(C(=O)NCC(CNC(c2cc(C(=O)OC)no2)=O)OC)cncc(C(C)C)c1 c1(C(N2CC(NC(c3ccc(OC)c(C)c3)=O)C2)=O)cc2ccoc2cc1F N1(C(C=CC(=O)N(C)C)=O)CCC2(CC1)CCN(C(C13CCOC1CCOC3)=O)C2 c1(SC)ncc(N)c(C(=O)NC(CNC(C2CNC(=O)N2)=O)CO)n1 CCCCC(CNC(=O)C(c1cccc(F)c1)OC)NC(c1ocnc1C1CC1)=O c1(C(N(CCCNC(C2(N(C)C)CC2)=O)C(C)C)=O)ccc(S(=O)C(C)C)cc1 C1(C(=O)Nc2cc(C(C)C)ncn2)CC12CCN(C(c1cc(C(F)F)no1)=O)C2 C1(CC(N2CC(CCNC(c3cnc(N(C)C)o3)=O)C2)=O)CC2(CCC2)C1 C=C1CCN(C(=O)CC2CCCCCC2)C(C(=O)Nc2ccc(F)cc2OC)C1 C1(C2CCCN(C(c3cc[nH]n3)=O)C2)(NC(c2cc(OC)ncc2Cl)=O)CC1 c1(CC)conc1C(=O)NC1CC(CNC(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(=O)NCC(C)CNC(C2(Br)CC23CCC3)=O)noc2c1COCC2 c1(C(=O)Nc2cccc(NC(C(C(C)C)C)=O)c2)cc(=O)cc(Cl)[nH]1 N1(C(CCn2c(C)nc(C)n2)=O)C2CCC1(CNC(=O)CC1CCCC1O)CC2 c1(C(=O)NCC(C)NC(c2cnc(C#N)s2)=O)ccc(S(C)(=O)=O)[nH]1 Cc1ccccc1S(=O)(=O)Cc1cnc(C2CCCC2)nc1O Cc1nn(CC(=O)NCC(C)(C(C)C)NC(=O)CCC2CCC2)c(C)c1C=NO C(=O)(C(F)(CNC(C1(C)CC1(C)C)=O)C(C)C)NCc1cc(OC)no1 CCC(CN(C)C)C(=O)NC(c1nocc1C(=O)N(CC(c1nn[nH]n1)C)C)C c1(C(=O)NCc2cnco2)cn2c(n1)CN(C(=O)Cc1ccc(Br)c(Cl)c1)CC2 c1(CC(C)N(C(c2ocnc2CC)=O)CC)nccn1C C1(C(COC)C)(C(=O)NCCC2CCN(C(=O)C(C)N(C)C)CC2)CCOCC1 N1(C(C(=O)N(C)C)=O)CCS(=O)(=O)C(CCNC(c2ccoc2Cl)=O)C1 CC(C)C(CNC(c1ccn(CCF)n1)=O)NC(=O)C(C)(C)c1ccccn1 S(=O)(=O)(c1ncccc1[N+](=O)[O-])N(c1ccc(C)cc1C)CC(C)C C=CC(CCC)CC(=O)NCCCCCNC(=O)C(C)(C)c1cccs1 C(=O)(C(C)(C)C(C)(C)O)NCCCCCCNC(c1cnc(C)nc1C1CC1)=O c1(OC)cc(C)cc(CNc2c[nH]nc2C(=O)N=c2cc[nH][nH]2)c1O c1(C(N(CC(C)NC(CC2CC(=C)C2)=O)C)=O)ccc(F)c(C)c1C c1(OC)ccc(CCN(C)C(=O)NCCC(C)CO)cc1OC(C)(C)C C1(C(=O)NC(C)(C(=O)NC2CCC3(CC3)C2)C2CCC2)CC2CCCC2C1 C1(NC(C2(NC(=O)CCc3cscn3)CCN(C)C2)=O)CC(F)(F)C1(C)C CC1(CNC(=O)COCC(F)F)CCN(C(c2ccc(C3CC3)cn2)=O)CC1 c1(C(=O)NCC(CN(C(C2CC(OCC)C2)=O)C)(C)C)cc(C)c(=O)n(C)c1 c1(CC(C)C)ncc(C(=O)NCc2cn(CCNC(=O)CCC3CC3C)nn2)[nH]1 C(C(CC)C(C)C)(c1nnnn1CCNC(N1CCC(C(CC)C)CC1)=O)NCC CC(C)C(CC(=O)NCCCCn1cc(CCO)nn1)c1ccccc1 C1(CNC(c2c(COC)ocn2)=O)CN(C(c2nnccc2C)=O)CC1O C1(NC2CCC(CNC(C(CCOC)C)=O)CC2)CC2CC(OC)C2C1 C(=O)(CC(C)(C)C)OC1CN(C(C(C)N2CCC2)=O)C1 C1(CCC(=O)NC2(CC)CC2)CCN(C(c2cc(C(N)=O)co2)=O)C1 c1(CC(=O)NCCOCCOCCNC(CC2CCOC2)CO)cn[nH]c1 N1(C(Cn2c(=O)sc(C)c2C)=O)CCC2CCN(C(c3ccnnc3)=O)CC2C1 C(=O)(C(CC(C)(C)C)OC)N1C(CC)C(C(N2CC(CC(C)(C)C)C2)=O)CC1 C(=O)(C(CC(C)C)NC)NC1CCCC(NC(N(C2CCS(=O)(=O)C2)CC)=O)C1 O=C(C1=C(Cl)CCC1)NC1CC(F)CN(C(=O)C(F)CC2CCOC2)C1 C1(CNC(C2CC(CCC)C2)=O)N(C(c2cnc(F)c(Cl)c2)=O)CCCC1(C)C c1(C(=O)Nc2ccc(NCCCC)cn2)ccn(CC)c(=O)c1 Cc1cc(C)c(C#N)c(N2CCC(OCCNC(=O)Cc3ccnc(O)c3)C2)n1 C(=O)(C(C(C)C)NC(=O)Nc1ccccc1)NC(C(C)(C)OC(C)C)C Cc1cc(O)ncc1C(N1CCC(CNC(c2occc2F)=O)C1C1CC1)=O N1(C(C2CC(CCC)C2)=O)CC2CC(C)N(C(=O)CC3CC=CCN3C)C2C1 CC1(C)CN(C(=O)C2=CCCSC2)CCC1C(NCP(C)(C)=O)=O c1(C(N2CCC(NC(C(C)CC(N)=O)=O)C(F)C2)=O)cc2n(n1)CCCO2 C1(C(=O)NCC2(C(C)(C)O)CN(C(c3n(CC)nnc3)=O)C2)CC(C(C)C)=NO1 Cc1ccnc(C)c1C(N1CC(NC(C23CCCC(C2)OC3)=O)CC(O)C1)=O CN1CCC2(CCN2NCCCC(F)(F)F)C1 C(CC(C(=O)NCC1CN2CCC1C2)NC(c1cnnc(O)c1)=O)OC C1(C(=O)NCc2ncccn2)COCCN1S(=O)(=O)Cc1ccc(Br)cc1 CC(C(C)(C)O)N(C(=O)C(O)C1CN(C(=O)Cc2cncn2C)C1)C C1(NC(COC(CC)C)=O)CN(C(c2cc(C)c[nH]2)=O)CC2(CCOCC2)C1 N1(C(C(C)=C2CC2)=O)CCC(F)(CNC(C2CCN(C)C2)=O)C1 c1(OC)nc(NC(=O)C(N2CCC(C)(c3cccc(F)c3)C2)=O)sc1C N1(C(=O)Nc2ccc(F)c(C)c2Cl)CC(N=c2ncnc3[nH][nH]c(Br)c2-3)C1 N1(C(CCC=C)=O)CCN(C(=O)CCCCC2CC2)C(C)CC1 C1(NC(C2CC2C(=O)N)=O)CCN(C(=O)C=CCN2CCC2)C1.C1(S)CC1 c1(CC)cc(F)c(C(=O)NC2CC(NC(C3CCCC(C)(C)O3)=O)C2)cc1F C(c1ccccc1)=CC(=O)NCC(C1CCCC1)NC(c1occc1Br)=O C12(C(=O)NCCOC3CCN(C(C(C)(C)OC)=O)C3)CCC(CC1)C2(C)C C1(C(CNC(CN(CCC)C)=O)(C)C)CCN(C(=O)Cn2nc(C)cc2N)CC1 c1(CC)c(C(=O)NCC2CC(NC(=O)C=Cc3cnc[nH]3)C2)cnn1C C1(C(C)C(=O)NCc2cccnn2)CCCN(Cc2ccns2)C1 C#CCC(CC(=O)N1CC(N(C)CC)C1)NC(C1CC(O)(C#C)C1)=O N1(C(C(C)SCC)=O)CC2CCN(C(C3CC(O)(c4ccncc4)C3)=O)CC12 C(=O)(C(C(C)(C)C)NC(C)=O)OCC(C1(c2ccon2)CCC1)C C12(C(=O)NCCCN(C(=O)CCc3cc(C)sc3C)CC)CC(C1)S(=O)(=O)C2 N1(C(C2(CC)CCCN(C(CC(CC)OC)=O)C2)=O)CC2CCC(C1)C2C#N N#Cc1ccc(NC(C2CC23CCN(S(=O)(=O)c2ccc(Br)s2)C3)=O)c(F)c1 Cc1nc(-c2cn(CC(C3CN(C(=O)CC4COCCO4)C3)F)nn2)sc1C c1(C(=O)NCCCN(C(c2scnc2C)=O)CC)ccc(C2CC2)c(C)c1 c1(N2CCN(Cc3cc(C(=O)OC)n(C)n3)C(C)C2)ncnc2occc12 c1(C(=O)NCC2C(NC(CCOC)=O)CCC2)c(C)coc1-c1ccccc1 Cc1ccnn1CC(=O)NCc1ncn(C(C)C)n1.c12nocc1C(=O)NC2C c1(C(=O)NCCC2CN(C(c3cn(CCOC)nn3)=O)C2)ncc(F)cc1F CC(C)CC(F)(F)C(=O)NCC1CCC(NC(=O)CCOc2ccc(F)cc2)C1 c1(C(=O)NC2(C)CCCN(C(=O)C(O)Cn3cncn3)C2)n[nH]c2c1COCC2 c1(C(=O)NC2C(NC(=O)OC(C)(C)C)CCCC2)cc(Br)c(F)cc1F N1(C(C2CCC(C)C2)=O)CCC(CNC(c2ccncc2C(=O)OC)=O)C12CC2 c1(OC)cc(F)c(C(=O)NC2CC2NC(c2c(C)n[nH]c2C)=O)c(F)c1F Cc1ccc(C(=O)NCC2COC(CNC(=O)NC(C)(C)C)C2)c(C)c1 Cc1occ(C(F)(F)F)c1CC(N1CC2CC2(NC(=O)CN(C)CCO)C1)=O C1(C)(CC(=O)NCC(C)N(C(=O)CN2CC3CC3C2)C)CCOC1 C(=O)(C(C#N)(CC)CC)NC(C=CC(N1CC(C=C)OCC1)=O)(C)C c1(NC(N2CCC(C(F)F)C2)=O)ccc2c(c1)OCCCO2 C(=O)(C(CNC(C1CCC(NC(C2CCC3(CC3)C2)=O)C1)=O)C(C)C)OC N1(C(C(CC)SC)=O)C(C(=O)NC2CCOCC2OC)CCC12CC2 c1(OCCC)cc(F)ccc1-c1nc(C(=O)NCc2ncn(C)n2)ccc1F C(N=c1[nH]c(=N)[nH]c(=NCC(F)(F)C(F)F)[nH]1)c1c(C2CC2)ccc(C)c1 c1(C(=O)NCC2(CNC(C3CCCC(O)C3)=O)CCC2)cccc2c1CC(=O)N2 CC1CC2CC(C(=O)NCCC(C)CCNC(c3cnc(O)c(Cl)c3)=O)(C2)O1 N1(CC(C)C)CCN(C(=O)CSc2ccccc2)CC1.C1(C)C(=O)N1 C(C(CCCC)NC(=O)CCOCCN(C)C)NC(C1(C#C)CCC1)=O C1(C(N2CCC(C#N)(F)C2)=O)CCN(C(=O)C=CC2CCOCC2)O1 CN=c1nc(C(N2CC3CC(NC(c4sccc4SC)=O)CC2C3)=O)cc(C)[nH]1 C1(C(N2CC(C)C(NC(=O)C3=CCCC3(C)C)CC2)=O)CCCC12CCOCC2 C1(=CC(=O)NC(C(C)NC(=O)C(C)(F)F)C)CCC(C)(C)CC1 CC1(C)CC(NC(C23COCC2C3)=O)CCN(C(C2(CC3CC3)CC2)=O)C1 c1(C(N2CC(C(C)NC(C3CS(=O)(=O)C3)=O)C2)=O)cc(Cl)c(N)c(Cl)c1 c1(CSCCC)ccc(C)o1.C1(C(=O)NCCN(C(=O)CN(C)CC)C)CCCC1 c1(-c2ccc(OCC)cc2)ccc(-c2nccn2C(C)CN(C)C)c(F)c1 CC1OC2(C)CC1(C(=O)N(C)CCN(C(=O)C(F)(F)C1CC1)C)C2 Cc1nc2c(o1)CCN(c1ncc(Br)cc1S(=O)(=O)NCC(C)(C)N(C)C1CC1)C2 C1(CCNC(C2CC(F)(F)C2)=O)CN(C(c2cc(C(F)(F)F)ccn2)=O)CCO1 c1(C(N(CCCNC(c2cc(Cl)ns2)=O)CCC)=O)ccc(CC)nc1C C(CN=c1nc2scnc2c(N2CC3CC3C2)[nH]1)c1c(Br)csc1 CC(C)(C)C(C#N)C(=O)NC1CC2CCC1C(NC(=O)COC1CC1)C2 Cn1nc(CC(=O)NCC2(CNC(=O)CC34COC(C)(C3)C4)CCC2)cc1Cl C1(n2ccnn2)CCCN(C(c2ncccc2F)C2CC2)C1 n1(CC)nnc(C(=O)NC(C)(C)C(C)NC(c2nnc(C(C)(C)C)s2)=O)c1C C(=O)(C(CCCOC)NC(c1ncc(F)cn1)=O)NC(c1ccn(C)n1)CC C(C)(C)(CC(F)C(=O)N1CC2CC1CN2C)NC(C(c1ccccc1)C)=O N1(C(C(CSC)O)=O)CC=C(C(=O)N2CCC2C(N)=O)C1 N(C(=NCCc1ccns1)N1CCCC(O)CC1)C(COC)C Cc1nccc(C(=O)NC(CNC(c2cc(-c3ccn(C)n3)on2)=O)CO)n1 C1(NC(C)=O)CCC(C(N2CC=CC(NC(=O)Cc3cnns3)C2)=O)CC1 c1(C(=O)NCC2CN(C(CCC=C(C)C)=O)C(C)CC2)c(F)ccc(C#N)c1F C1(NC(C(N)=O)=O)COCCC1NC(c1cccn1C1CC1)=O C1(N(C(CCC(C)OCC)=O)C)CN(C(=O)Cn2ccc(O)nc2=O)CC1(C)C Cc1cc(C(=O)NCC2(F)CC(NC(C34CCCC3C4)=O)C2)c(C)n1C1CC1 c1(CC)cccc(CC(=O)NCC2C=CCN2C(c2cnn(CC(C)C)c2)=O)c1 C(C(CC(C)C)NC(=O)CC1CC2CC2C1)NC(c1ncn(CC)n1)=O C1(CNC(CCCSC)=O)CCC2(CN(C(=O)CC(C)(F)F)C2)O1 C(C(=O)N1CCCCC1CC(F)(F)F)(C(C)(C)C)n1cc(CCC(C)O)nn1 N1(C(C(CC=C)C)=O)CCN(C(C2CCCOC2)=O)CC12CC2 C(C)(CO)(C(=O)N(CCCN(C(=O)CC(c1c(C)noc1C)C)C)C)OC C1(C(N2CC(C(=O)N(CCO)CC3CC3)(OC)C2)=O)CCC2CC1CO2 N1(C(C(C2(O)CCCCC2)NC(CC2C(C)(C)OCC2)=O)=O)CC2CC1C1CC21 CS(=O)(=O)C1CC(C(N2CCN(C(=O)COC(F)F)CC2c2ccccc2)=O)C1 C(=O)(C(O)C(C)C)NCC(=C1CN(C(CCc2ncc(C)[nH]2)=O)C1)F C#Cc1ccnc(C(=O)NCC(CC)NC(c2ccon2)=O)c1 N1(C(C2C(C)C2)=O)CCC2(CC1)CN(C(C1CNC(=O)CC1C)=O)CCO2 C(=O)(C1=C(Cl)CCOC1)N1CCCC(COC)C1.c12occc1CNC2=O c1(C(N2CC(CCNC(C(C)=C3CCC3)=O)OCCC2)=O)cc(C)c(C#N)cn1 CC1C(C)N(C(CCC)=O)CCN1C1CC1c1c[nH]c(-c2nn[nH]n2)c1 CC(C(=O)N1CC(NC(c2ccc(CCC(N)=O)cc2)=O)C(C)C1)S(N)(=O)=O C1(CNC(c2c(SCC)cccc2)=O)CN(C(c2cc(C)no2)=O)CC12CCC2 CC1CCC(CC(N2CC(C)(NC(=O)Cc3ccn(C)c3)C2)=O)OC1 Cc1ccc([N+](=O)[O-])cc1C(N1CCCC(C(N)=O)C1)=O CC1(C)CCC(C(N2CCCC2CNC(c2cnc(=N)[nH]c2)=O)=O)C1 CCC(C)(CNC(C)=O)C(=O)N1CC2CC1CN2C(=O)Cc1n[nH]c(C)n1 C12(C(=O)OCC)CC1CCN2Cc1csc(N2CCCCC2)n1 c1(C(N2C(CNC(C3(C(C)C)CCC3)=O)CCC2)=O)cc2c[nH]cnc-2n1 C1(NC(C(CC)C)=O)CCC(C(=O)N(C)Cc2ccccc2OC)CC1 c1(C(=O)NC2(CCNC(c3ncn(C)c(=O)c3)=O)CC2)cc2c(nn1)CCCO2 C1(C2CCCN(c3cc(C#N)nc(C4CC4)n3)C2)(NC(C2(C)C=CCC2)=O)CC1 c1(C(=O)OC)cc(C(=O)NC2CN(C(=O)CC(F)(F)F)CCC2CO)c(F)cn1 N1(C(C=Cc2c(OCC)cccc2)=O)CCCN(C(=O)CCC2(C)CC2)CC1C CN(CCN1CCOC1=O)N1CCC(c2ncc3n2CCOC3)CC1 C1(NC(CCNS(CC)(=O)=O)=O)CCN(C(=O)CC2(N(C)C)CC2)C(C)C1 C1(NC(C2C(CC)N(C(=O)CC3C(=O)NN=C3C)CC2)=O)CC2(C1)CC(C)C2 C1(NC(c2c[nH]nc2C(F)(F)F)=O)CC2CC1N(C(=O)Cc1cnc[nH]1)C2 c1(C(=O)NC(C)CNC(c2cc(C3CC3)cs2)=O)ccc(=O)n(CCO)c1 N1(C(C(c2ccnn2C)C)=O)CC(C2CCCCN(C(=O)C(=O)NC3CC3)C2)C1 c1(C(N2CCN(c3ccn(C)n3)C3CC23)=O)cnc2ncccn12 c1(C(N2CCC(C(=O)NCC(C#C)OC)(C(C)C)C2)=O)cncc(F)c1C c1(-n2cc(C(C)(C)NC(c3nc(CC)sc3)=O)nn2)ccc(F)c(Cl)c1 C(=O)(CCC(=O)NC1CC1CNC(c1cnn(CC)c1Cl)=O)NCCC C1(C(N(C)Cc2cnc(C)s2)=O)CC2C=CC1N(C(c1cnns1)=O)C2 c1(CC(N2CC(N(C(c3nc(CCC)sc3)=O)C)C2)=O)ccccc1C(F)(F)F C1(C(N2CCC(C)N(C(c3nc(Cl)cs3)=O)CC2)=O)CCCC2CCCCC12 C(c1c[nH]c(=N)c(C)c1)=CC(=O)NCC(C1CC1)NC(c1nnn(CC)c1C)=O Cc1c(Cl)ccc(C(=O)NC2CC2C(=O)Nc2cccc(F)c2C#N)c1Cl C(C(=O)Nn1cnn(C)c1=S)(C1N(C(COC)=O)CCC1)OCCCC Cc1nn(C)c(NCC2CC(=O)N(CC3CC3)C2)c1C#N C(=O)(C(CCOCCO)NC(C1CCC(=O)N1)=O)OCC N1(C(C(CC=C)NC(C)=O)=O)CCN(C(c2cc3n(n2)CCC3)=O)CC1C(F)F C1(NCC(C)CC(F)(F)F)(NC(=O)OC(C)(C)C)CC(C)(C)OC(C)(C)C1 N1(C(c2nc(C(C)C)oc2)=O)CC(C)CN(C(=O)CCC2CCCN2C)CC1C C1(C)(CNC(CN(C(=O)C(C)OCC)CC#C)=O)CC2(CCC2)C1 CC(C)C(F)C(=O)NC(c1nocc1C(=O)NCC1CC(CN(C)C)C1)C C1(C(N(CCCCN(C)C(c2cc(C3CC3)on2)=O)C)=O)CCOCC1(C)C CCC(CCC(=O)NCC1CCCN1C(=O)C1=C(C)CCC1)OC Cc1oc(CCN)nc1C(=O)N(C(C)Cc1cccc(Cl)c1)C N1(C(c2c(CC)nccc2)=O)CCCC2(NC(=O)C(C)CC(C)(C)C)CCCC12 N1(C(C2(c3ccc(C)cc3)CCC2)=O)CC(CNC(C2CC2(C)C)=O)CC1(C)C C1(CCNC(C(COC)NC(C)=O)=O)CSCCN1C(=O)CC1CCCOC1 c1(C(=O)NCC(CC=C)NC(=O)CCC2CC2(C)C)ccc(C(C)C)nc1C c1(CC(=O)NC(c2ccc(F)c(F)c2)(C(=O)OC)C)cccc2c1CCC2 C1(OC)(CNC(=O)C(F)n2ccnc2)CN(C(=O)CSCc2cccs2)C1 c1(C(N2CCN(C)C(CNC(C3CC4(CSC4)C3)=O)C2)=O)cc(N)c(O)c(F)c1 CN1C(=O)OCC12CCN(C(c1cc(C(=O)O)c3n1CCCC3)=O)C2 C1(C(=O)NC(C)C(c2ccccc2)NC(c2cncc(F)c2)=O)CCN(C)CC1 C#Cc1cccc(C(C(=O)NCCCCC=C)NC)c1.C1(C#N)(COC)CC1 CCCC(CCCNC(c1ccc(-c2ncc[nH]2)nc1)=O)NC(=O)CCCC#N c1(C(=O)NCC2(F)CCCN(C(C3(CC#C)CCC3)=O)C2)cccc2ncsc12 c1(C(N(CC(C)NC(c2c(OC)c(C)sc2)=O)C)=O)cc(OC)nc(F)c1 C(C(C)(O)CC(=O)N1CC(NC(=O)Cn2cnc(C(N)=O)n2)CC(F)C1)OC CCC(CCCC(=O)N1CCC1C(C)O)NC(=O)C1=C(C)OCC1 c1(N(CC(=O)NC2CC(NC(C3CC3(C)C(F)F)=O)C2)C)ccc(Cl)cc1 c1(C(N2CC(C)CC(NC(CCSC)=O)C2)=O)cncc2ccccc12 C1(CC(=O)N(C2CCCN(C)C2)C)C2CCCC2N1C(=O)CC1CC2(CC2)CO1 O=C1OCCCN1Cc1cn(CC(=O)N(C2CC2C2CCC2)C2CC2)nn1 c1(C(=O)OCc2ncc(-c3ccc(Cl)cc3)o2)cccc2cc(O)ncc12 c1(OC)nc(C(=O)NCCCNC(=O)C(C)c2ccco2)co1 N1(C(CCCCC)=O)CCCCC(C2CN(c3nc(Cl)nc4c3SCC4)C2)C1 C(=O)(C(C)C(C)(F)F)N(CCNC(CC1CC(NC(C(C)C)=O)C1(C)C)=O)C C1(C(N2C(C=C)COCC2)=O)N(C(C2OCCOC2C)=O)CC12CCCC2 Cc1cc(C(=O)NCC2C=CCN2C(=O)C(C)n2cnnn2)c(C)cc1Br c1(C(=O)NCCN(C)C(C2(Cl)CC2(C)C)=O)ccccc1C(C)(C)C C1(CNC(C(N2CCC(C(C(=O)OCC)C#N)CC2)=O)=O)COC2(CCC2)C1 N1(C(c2nc(C)sc2)=O)CC(CNC(c2nnn(C)c2C(F)(F)F)=O)CC1C C1(CNC(CCc2nc(C)c(C)o2)=O)CN(C(=O)CC2CC2(Cl)Cl)CC12CC2 C(=O)(CC1=NNC(=O)C1)NC1C(NC(CC(CC)CC)=O)CCCCC1 Cc1cc(C)n(CCNC(=O)CN(C(C2CC(O)C(F)C2)=O)C2CC2)n1 c1(C(N2CC(n3cc(C(CC(C)C)O)nn3)C(C)C2)=O)noc2c1CCCC2 Cc1nc(C(=O)NCCC2=CCN(C(=O)CN(C)CCO)CC2)c2ccccn12 c1(C(=O)NCCN(C(c2cc(C)cc(C#N)c2)=O)CC)cc2ccncc2cc1F N1(C(c2cc(OC)no2)=O)CCOC2(CCCN(C(C3CC(C)(C)CO3)=O)C2)C1 CCCC(C(=O)NC1CC(C)N(C(=O)Cn2cnc(=N)[nH]2)C1)OC c1(CC)noc(C2CCC(NC(=O)CC3(OC)CCOC3)C2)n1 S(=O)(=O)(c1nc(N2CCC(N(C)C)C2C)ccc1Br)NCC1ON=C(C)CC1 C1(C2CCCCO2)(C(=O)Nc2c(C)nn(CCF)c2)CCCO1 Clc1ccc(C(C2CC2)NCc2nnc(C3CCCCC3)s2)cn1 Cc1ccccc1C(=O)OC.c1(C2C(=O)NC(C)CN2C)ccc(C(F)(F)F)cc1 C#CC1CCCN(C(C2CCC(CNC(C3CCC(CC)CC3)=O)CC2)=O)C1 c1(C(=O)NCCC2(CNC(c3cnc(CC)s3)=O)CC2)c(F)c(F)c(F)cc1F N1(C(C2CC=CCN2C(=O)COCC2CC2)=O)CCCC(F)(F)CC1 C12CCCCC1OCC(=O)NC2.CC(C)CCNC(=O)C(=O)C1CCCC1 N1(C(C(C(C)C)N(C)C)=O)CCC2(C1)CN(C(c1ccco1)=O)CC(C)O2 N1(c2ccc(C#N)cn2)CCC2(NC(c3ccc(C4CC4)o3)=O)CCCC12 CC(C)(CC(=O)NCC(CNC(C1CCCSC1)=O)CO)C1CC1 CCCCCCCCCCCCn1cc(C(=O)NC2CC(C(=O)OC)C2)nn1 C1(OC)CN(C(C2(C)COC(=O)C2)=O)CC1NC(c1cc(C)nn1CCO)=O CCC(CCOC)C(=O)NC1CC(N(C(=O)CSCCC(F)(F)F)C)C1 C1(NC(=O)CC2CC=CC2)CN(C(=O)CCSc2ccccn2)CC12CCC2 Cc1cccc(C=CC(=O)NCCCCC(C)NC(c2cnc(C(C)C)[nH]2)=O)c1 C1(C(N(CCNC(Cc2nc(CC)sc2)=O)CC)=O)CCc2nc[nH]c2C1 c1(C(=O)NCC(CNC(C(CC)N2CCCC2=O)=O)(C)O)cc(Cl)cn1CC c1(C(C)C)ccc(CC(=O)NCC2CN(C(C3CC3C(N)=O)=O)CCO2)cc1 C1(C(N2CC(N(c3cc(=O)n(C)cn3)C)C2)=O)CCC2CC2CC1 C1(C(=O)N(CCCN(C)C(C2CCC3(CCC3)C2)=O)C)(OC)CCC(C)(C)C1 CCC(C)C(=O)C(=O)N1CC2CC(C1)N2C(=O)CC(C)(C)C1CC1 c1(N2CC(C(C)NC(CCCC)=O)OCC2)nc(C)nc2scc(C)c12 N1(C(C(C2CCCC2)NC(c2nc(COC)oc2)=O)=O)CCC(C)(C)CC1 C1(C(F)F)(CNC)CCN(C(c2cnccc2C)=O)C1.c12ccnc(c1)OC2=O CC1CN(C(C2CCCC3CC23)=O)CC1CNC(=O)C(c1ccccc1)(C)N(C)C N1(C(C(CCC)CC)=O)CC(C)(C)OCC1CNC(c1ncnc(O)c1F)=O c1(C(N2CCCCC(NC(Cc3cc(C)on3)=O)C2)=O)cc2cc(F)ccc2o1 c1(C(=O)NC2CCN(C(C(CC)=CCCC)=O)C2)ccccc1SC(F)F N1(C(c2c(N)cc3c(c2)CCC3)=O)CCC(C2CCCN(C(=O)CC(F)F)C2)C1 Cc1[nH]nc(CNC(C2CSCN2C(=O)CCOCC2CC2)=O)c1C c1(CSCC)ncccc1C(=O)NC(C1(CNC(C)=O)CC1)C N1(C(C2C(C)C2)=O)CCCC2C1CCCN2C(c1cccn(C)c1=O)=O c1(C(=O)NC2(CCCCNC(CC(=O)NCC)=O)CC2)ccccc1OC C1(C2CCC2)(C(=O)NC(C(C)NC(=O)CCc2n[nH]c(C3CC3)n2)C)CC1(F)F c1(C(=O)NC2CC2CC(N2CC(OCCC(=O)NCC)C2)=O)cncc(C)n1.C(O)C n1(CC)cc(C(=O)NC(C2CCN(c3ccc(C(F)(F)F)cn3)CC2)C)c(C)n1 Cc1cc(=O)c(C(N2CCC23CCCCC3)=O)nn1-c1ccc(F)cc1 c1(OC)ccc(Br)cc1NC(C12CC1CN(Cc1ccc([N+](=O)[O-])s1)C2)=O C1(C)(C(=O)NCC(C)NC(c2ccncc2Cl)=O)CC(C)(C)C1 N1(C(c2n(C)[nH]c(=N)c2)=O)C2CCC1CC(NC(C1CC3(CCCO3)C1)=O)C2 C1(OC)CN(C(=O)CC2CC2(Cl)Cl)CC1C(=O)NCC=CCSC c1(OC)cc(C(=O)NCC(O)CCNC(C23CCCC2(C(N)=O)C3)=O)ccc1C C(CCCC(CO)NC(C1C=CC=CC=C1)=O)NC(C(C(C)O)N(C)C)=O N1(C(C(CC)SC)=O)CCSc2ccccc2C1 CCC(CC(=O)N1CCC(CC)C1CC)NC(C)=O.C1(=O)CC2(CC2)N1 CCCCC(O)C(=O)NCCCC1CCCCN1C(c1[nH]nnc1C)=O Cc1cc(C(=O)NCC(C)(CO)NC(c2csc(Cl)n2)=O)nc(O)c1 CCC(C)C(O)C(=O)N1CC(CC(C)NC(C2CC3(CCOC3)C2)=O)C1 C1(NC(c2c(CC)occ2)=O)CCN(C(c2nc(C)ccc2C)=O)C(C)C1 c1(N(C2CC3CNC2C3)C(C(C)n2cncn2)=O)ccc2cc[nH]c2c1 C=CCC(C(=O)NCC1(O)CCCN(C(c2cc(C3CC3)on2)=O)CC1)C(C)C c1(C(c2n(CCC)nnn2)NCc2ccc(Br)c(Br)c2)sc2ccccc2c1Br c1(CCOCCOCCC(=O)N)ccc(P(C)(C)=O)o1.C1(C(CN)C)(OCC)CC1 c1(C(C)(C)C)nc(CC(=O)NC2CC(C)(NC(c3n[nH]cc3Cl)=O)C2)cs1 N1(C(C2C(OCC)C2)=O)CCSCC1CCNC(c1cnc(C2CC2)o1)=O C1(C(N2CC3C(NC(c4cc(C)[nH]n4)=O)C(C3)C2)=O)Cc2ccccc2C(=O)O1 c1(CC(=O)NC2C(NC(c3c(CC)scc3)=O)CC2)ccc(-n2cnnc2)cc1 C(=O)(C(F)CC(C)(C)C)N1CC(C)N(C(=O)Cc2cnoc2)CC1 C1(NC(c2ncc(C)cn2)=O)C(C)CN(C(=O)CCc2cn[nH]c2)CC1C N(C1CCc2c1ccc(Cl)c2Cl)C(Cc1cccc(OC)c1)(C)C1CC1 CCC(F)(C(=O)OC)C(=O)N1CCC(NC(=O)COC(C)C)C(F)C1 C1(CNC(C(C)n2ccnn2)=O)CCC(NC(=O)CCc2ccncc2)CC1 c1(OCC)nc(N2CC(CNC(C3CC3C3CCCCC3)=O)C2)ns1 C=C=C(C)CC(=O)N1CCCC1C1CC1.C1(C(=O)OCC)CCCO1 CC1CCCC(C)N(C(C2(N=[N+]=[N-])CCN(C(C3CCSC3)=O)C2)=O)C1 C(=O)(C(C)CC(=O)NC1CN(C(=O)C(C)N(C)C)CC1(C)C)OC C1(NC2(OC)CC(C[Si](C)(C)C)C2)CCCC1(C)C C(=O)(CCCCC(C)(C)C)N1CC(OC)(CNC(=O)CCc2cccc(O)n2)C1 C1(C)(C(=O)Nc2ccc(N(C)C)cc2)CCCN(Cc2ccc(Cl)c(Br)c2)C1 Cc1c(CC(=O)NC2CC2NC(=O)Cc2cccnc2)ncn1C N1(C(c2c(C)nc(C3CC3)s2)=O)C2CCC1CN(C(C1CCC(CO)CC1)=O)C2 N1(C(Cc2cccc(C(C)(C)C)c2)=O)CC2COCC(C1)C2NC(=O)C(N)=O C1(C(=O)NCCOCCCOCC(F)F)(OC)CC(NC(=O)C(O)C2CCC2)C1 c1(OC)cccc(C(N2CCC3C(NC(C4CCCS(=O)(=O)N4)=O)C23)=O)c1OC c1(N(C)CC2N(C(c3c(C)nc(C(C)C)o3)=O)CCCC2)ncn(C)c(=O)c1Br c1(C(=O)NC(C2CN(C(c3ccc(CO)o3)=O)C2)C)ccc2cncn2c1 N1(C(c2cc(COC)no2)=O)CCC(CNC(=O)CC2CCNC2=O)C12CCC2 C(=O)(CCCS(=O)(=O)N1CCCC1)N1C(C)CN(C(C2OCCC2(C)C)=O)CC1 c1(C(C(=O)NCCN(CC(C)O)C(c2ccsn2)=O)OC)c(F)cccc1F c1(C(N2C(C(=O)NCC3CN4CCC3C4)(CC)CCC2)=O)cc(CO)cc(F)c1 c1(C(N(C2CC(NC(C3C(=C)C3C(=O)OC)=O)C2(C)C)C)=O)nc(C)ccc1OC N1(CC(=O)Nc2ncc(C(C)=O)s2)CCCNC(=O)C1(C)C C(C(C)(C)C(=O)N1CC(N(C)C)C(F)C1)N(C(CCC1CC(C)C1)=O)C CC(C)(CCCF)NC(=O)C(C)(CO)NC(c1cnc(C(C)C)o1)=O c1(C(=O)NCCN(C(c2cc(C(C)C)no2)=O)CC)cn(C)c(C)c(Br)c1=O CC1(C)C(CNC(=O)C(N)=O)CCN1C(=O)CC(=O)NC1CC1 Nc1cccc(F)c1C(=O)NCCC1(CNC(c2ccc(N)cc2)=O)CC1 c1(C2C(Cl)C2)nc(C2CCCc3ccccc32)nn1C1CCSCC1 Cc1ncc(C(=O)NC(C2CCCN2C(=O)C(F)C2CCCC2)C)o1 C1(F)(CNC(c2cc(C)n(CCO)n2)=O)CCCN(C(c2cnc[nH]2)=O)C1 c1(CCC(=O)NC(CC)(CNC(C2C(C)C2C)=O)CC)ccccc1[N+](=O)[O-] C1(C(C)NC(=O)COCP(C)(C)=O)CCN(C(=O)CNS(C)(=O)=O)CC1 c1(C(=O)NCCCC(C)NC(CCc2cc(C)no2)=O)cc2c(s1)CCCC2 C1(C)(C(=O)NCc2c(C(=O)NCCC3(CN(C)C)CC3)nco2)CC(C)(C)C1 Cc1cc(C(N2CC(F)(c3cn(C(C)(C)C)nn3)C2)=O)cc(C)c1Br C1(C(=O)NC2CN(C(C(CC)=CC)=O)CC2C(F)(F)F)CC2(C1)CC21CCC1 N1(C(C2CC(C)OC2)=O)CCCC(C)(C)C1CNC(=O)CC1NC(=O)NC1=O CCC(CC(=O)N1CCCC(CN(C)C(C2CCC2OC)=O)C1)C(F)F O=C(CCCCCCCCC1CC1)NCCNC(c1cnc2c[nH]nc2c1)=O N1(C(c2c(C)ncs2)=O)CCCC2(CCN2C(c2[nH]cnc2C#N)=O)C1 N1(C(c2cc(C)nc(O)c2)=O)CCCC(C2CC2NC(=O)C=CC2CCOC2)C1 CCC(C(=O)N1CCC(CNCc2ccccc2Cl)C1)C(C)C c1(OCCC)ccccc1C(=O)NC(C)CNC(=O)CCC1CCCC(=O)N1 CC1CN(C(=O)CC2CC3(CCC3)CO2)CCCN1C(c1ccccc1Br)=O Cc1[nH]nc2c1CCC(C(=O)Nc1c(Br)ccc(F)c1F)C2 C1(NC(C(N)=O)=O)(CNC(=O)COCCOCCO)CCCCC1 C(=O)(C1(C)COc2ccccc21)NC(C)CN1CCN(C(=O)CC(C)(C)C)CC1 c1(C(N2CCCC(C3OCCO3)C2)=O)cn(C2CC2)nc1-c1ccccc1 CC1(C)CCN(S(=O)(=O)N2CC(c3ccc(F)cc3F)C2)CC1 N1(C(C2C(OC)CC2)=O)CCC(c2cc(CNC(C3CC34CC4)=O)on2)CC1 c1(CCNC(C2(c3cccs3)CCOCC2)=O)ccc2cccnc2c1 C1(N(C(=O)CSc2nc[nH]n2)C)CCCN(C(=O)COCC(F)(F)F)C1 c1(C(N2C(C(=O)NCC(C)OC)CC(F)(F)C2)=O)cc(I)c(F)cc1F c1(CCNC(C2CC(n3cc(CC(CC)C)nn3)C2)=O)ccc(C)cc1C C1(C(N)=O)CCC(CC(N2CC(=CCNC(=O)C(O)CN3CCCC3)C2)=O)CC1 C(=O)(C(CCC1CC1)NC(c1cc(C)co1)=O)NC(CCOC)CNC(C)=O N1(C(C2C(CC)CCC2)=O)CCN(C(c2cnn(C(C)(C)C)c2N)=O)CC1C C1(C(=O)Nc2cccnc2)(CC)CCN(C(c2cccc(CO)c2)=O)C1 N1(C(C2CN(C(C)=O)C2)=O)CC2CCOCC2(NC(c2ccc(C)s2)=O)C1 C(=O)(C1=CCC(NC(c2nc[nH]n2)=O)C1)NC(C(=O)OC)C1CC1 N1(C(c2c(N)cncc2)=O)CC2(CCCC2)C1C(N1CCC2(CCC2)C1)=O N1(C(Cc2n(C)nnc2)=O)CCC2CCC(NC(C3CCCC(C)(C)C3)=O)C1C2 Cc1cc(C(N)=O)cc(C(=O)NC2(CCNC(c3cscc3C(F)F)=O)CC2)c1 C1(C(=O)NC2CN(C(C3(C)CC=C(C)CC3)=O)C2)CCN2CCCC2C1 C(CCC(O)C(=O)N=c1cc2ccccn2[nH]1)NC(c1cc(CC)oc1C)=O N1(C(C(CCCC)NC(=O)CC2C(=O)NN=C2C)=O)CCC(O)C(C)(O)C1 C1(CC#C)(NC(=O)NCC(c2ccnn2C)O)CCCCC1 c1(C(=O)NC(C2CCOC2)CNC(c2ccc(OC)o2)=O)nc(C)ccc1C c1(C(N2CCC(OCC#C)C2)C(=O)NCCC#N)cccc2occc12 C1(C(=O)NCC2(O)CN(C(CC3C(C)(C)C3)=O)C2)CCn2cncc2C1 C(=O)(C(C)(C)NC(=O)OC(C)(C)C)NC(CC)CNC(c1cnno1)=O c1(NC(C2N(C(C3CC=C(C)CC3)=O)C3C(C2)C3)=O)cc(Cl)c(O)c(Cl)c1 n1(CC(=O)N(C2CCN(C(C3CC3F)=O)C2)CCO)cc(C(F)(F)F)nn1 c1(NC(C2N(C(CC(CC)O)=O)C3C(C2)C3)=O)ccnc2cc(Cl)ccc12 C12(NC(c3c[nH]c(=O)cn3)=O)CCCN(C(C3CC(OC(C)(C)C)C3)=O)CC1C2 C1(O)(CNC(CCNC(C)=O)=O)CCN(C(=O)CCc2ncccn2)C1 C(=O)(C1=CCC(C)(C)CC1)NC(CCCOC)C(=O)NC(C)CSC C(=O)(C#CC1CCOCC1)NCCSC.O=C(CCCOc1ccccc1)Nc1ccccc1 C=CCCC(F)(F)C(=O)NCC(O)CNC(c1ccnc(SCC)c1)=O C12(C(=O)NC3CN(C(=O)C=Cc4cccc(F)c4)CC(F)C3)CCC(CC1)CC2 C(C(CC(F)(F)F)OC)NC(=NC)NC(c1ccn(C)c1)C N1(C(CN(c2ccncc2)C)=O)C(CNC(C2CC(C)(C)CO2)=O)CC2CCCC12 c1(C(=O)NCc2cc3n(n2)CCC3)nc2ccc(-c3cccc(O)n3)cc2s1 C12(C(=O)NC3CCC(NC(=O)CCc4cccnc4)CC3)CSCC1C2(F)F c1(CCOCC(=O)NCC(CN(C(=O)CCc2cnn(C)c2)C)O)ccccc1 c1(C(=O)NC(CNC(c2cn(CCC)nc2)=O)C)nccn2c(C)nnc12 c1(CNC(Cc2cc(C)sc2)=O)ccc(CNC(c2cnsn2)=O)cc1 C1(NC(C=CCCC)=O)CCS(=O)(=O)C12CN(C(c1nc(C)ccc1C)=O)C2 C1(C(=O)NCC(=O)OCC#C)C2CCC(C2)C1NC(c1cn(C(C)C)nn1)=O Cc1nccc(CN(C(=O)CCCn2cc(CO)nn2)C)n1 c1(C(C)=O)ccncc1.C1(C(=O)N)CCCC(C(=O)O)C1 CC1(CCNC(C2CC2F)=O)CCN(C(c2ccc(N)cc2O)=O)CC1 c1(C(=O)OC)ccc(C(=O)NC2(C)CCC(NC(=O)CN3CCCC3)C2)nc1C c1(NC(=O)OC)ccc(NC(C2C=CC(NC(c3ccnnc3)=O)C2)=O)cc1 Cc1cncc(C(N2CC(=O)CC2C(N2CCC(CC(F)F)C2)=O)=O)n1 Cc1noc(C)c1S(=O)(=O)NC1CCN(Cc2n[nH]c3ccccc23)CC1(C)C CC1CN(C(=O)CNC(=O)C(C)(C)C)CC1(C)CNC(=O)CSS(C)(=O)=O c1(C(=O)NCC2(COC)CCN(C(=O)COC(C)=O)CC2)cc2cccnc2[nH]1 Cc1cc(C(=O)NC2(CCNC(=O)C(C)(Cl)Cl)CCC2)sn1 C1(N(C(=O)C=C(Cl)Cl)CC)CC2CCC(C1)N2C(C1(C(F)F)CCCC1)=O c1(C(=O)NCC2OCC(CNC(c3csnn3)=O)C2)ncc(Cl)cc1Cl c1(NC(C(C(CC)CC)OC)=O)ccc2c(c1)CN(C(=O)COCC(F)F)C2 c1(CC)cc(C(N2CCC(NC(=O)COCC3CCCOC3)CC2)=O)ccc1Cl N1(C(C(CC)OCC)=O)CC(C)(CNC(=O)Cc2ccn(C)c2)CC1(C)C N1(C(C=CCCC(C)C)=O)CC(C)N(C(=O)C#CC2CCOC2)CC1C C#CC1CC2(CC2)CN1C(c1cc(CNC(c2ccc(C#N)cc2)=O)ccn1)=O Cc1[nH]c(C#N)cc1C(=O)NC1C2CC(NC(C3CC3C3CCC3)=O)CC12 N(C1COc2ccc(Br)cc21)C(=O)Nc1cccc(C2(C(F)(F)F)CCC2)c1 C(C)(C(=O)C(C=C(CN(C)CCO)C)=O)OCCNCC(F)F.CO.OC C1(C(C)C)C(C(C)C)CN1C(=O)CCOCCCNC(C1CC1Cl)=O.C(C)(=O)O CCCC(C)CC(=O)N1CC(O)(C(F)C(=O)N(C)CCc2ccccn2)C1 C(=O)(C1=NOC2COCC12)N1CC2C(N(C(c3c(N(C)C)nccc3)=O)C)C2C1 CC(C)(O)CC(=O)NCc1cccc(CNC(=O)C(C)(C)c2cccs2)c1 C1(CCCn2c(N(C)OC(COC(C)C)C)nnn2)CC(C2CC2)=NO1 N1(C(=O)OC)CCC(C(=O)NC2C3CC2N(C(=O)CCCOC(C)=O)C3)CC1 CC(C)CCC(O)C(=O)NC1COCCC1C(N1CC2(CCOCC2)C1)=O C1(N(C(c2cn(CC)nn2)C(=O)NC2CCC2)C)(SC)CCOCC1 c1(N(C2C(NC(=O)OC)CCCC2)C)nc2ccccc2s1 N1(C(c2c(C(C)C)noc2)=O)CCC(NC(=O)CCN2CCC2)CC(C)(C)C1 c1(C(=O)NC2CCCCN(C(c3ncc(C)cc3F)=O)C2)nc2cnccc2s1 C1(OC)C(OC)CN(C(=O)C(C(C)C)c2cc(C)no2)C1CNC(=O)C(C)C CC(C)C(F)(CNC(C1CCCO1)=O)C(=O)NCCCc1nncs1 CC1CCc2c(C(=O)N(CC(O)CNC(=O)C#CC3CC3)C)csc2C1 CCCC(C)CC(=O)N(CC(=O)NCCOC(C)=O)C.C1CC(=O)N1 C1(NC(c2cccc(C)c2)=O)CC2(C1)CC(NC(=O)CC1CCCNC(=O)C1)C2 C#CC(CNC(C1(NC(=O)C(C)C2CCC2)CC(CO)C1)=O)C(C)C CCCC(C)CC(=O)NCC12CC(NC(=O)Cc3ccn(CC)n3)(CCO1)C2 N1(CCCOC(C2(c3cccc(F)c3)CC2)=O)CC2CCC1C2 C1(C(=O)NC2CCC(C)N(C(=O)C(C)(C)F)C2)CCc2ccnn2C1 Cc1cc(N2CC(C)C(C)(CO)C2)nc(=NCc2cc(C(N)=O)co2)[nH]1 N1(C(C2N(C)CC(C)(C)C2)=O)CC2CCCC(N(C)C(C3CCCSC3)=O)C2C1 C1(C(=O)NCC(C)(C)CC2CCC2)CCCC(O)C1 c1(OC(C)C)nc(N2CCN(C(c3nc[nH]n3)=O)C(C)C2)ncc1Br C1(NC(C2CC(C)CN2C(c2ccccc2C#N)=O)=O)CC2(CCCC2)C1 C(C(=O)N1CCC(NC(C2CC2(F)F)=O)C1)(C(C)C)NC(=O)OCC c1(C(N2CCC(NC(c3c(CCC)n(CC)nn3)=O)C2)=O)cc(F)cc(F)c1F N1(C(C2C(=O)NC(=O)N2)=O)CCC(C2(NC(=O)CCC3CCCCC3)CC2)CC1 Cc1cc(CCNC(C23CC(NC(=O)CC4COCCO4)(C2)C3)=O)on1 C1(C(N2CCC(CC)CC2)=O)CCN(C(c2csnc2OC)=O)C1(C)C C(=O)(CCCCCS(N)(=O)=O)N1C2CN(N3C(C=O)CCC(C)C3)C(CC2)C1 C(=O)(C(C)(C)CCNC(=O)C=CC(=O)NC(C)C)N(CCN(C)C)C c1(C(=O)NC(CC(N)=O)C2CC2)ccccc1NC(c1ccc(Cl)cc1)=O C1(CC)C(C)CCCN1C(C)=O.N12CC3CC1CN3c1nnnn1CCCO2 N1(C(C=CC(C)(C)C)=O)CC(NC(c2cccc(C3CC3)c2)=O)CC12CCOC2 C1(NC(=O)CCC2CCCCC2)CCCCC1CNC(c1nsnc1O)=O c1(C(N2CCCC(NC(C(CC)(C)F)=O)C2)=O)cnc(C2CC2)nc1O Cc1cc(=NC(=O)C2CCN(C(=O)CC3CCCN3C)CC2O)[nH]n1C(C)C C(=O)(CCCCC(C)(C)OC)N1CCN(C(C2CCC(CC)CC2)=O)CC1CC C1(C)(C(=O)NC(C)CCCNC(c2c[nH]cc2C2CC2)=O)CCC(C)C1(C)C C12(C(N3CC4C(CO)C4C3)=O)CC3CC(CC(C3)C1)C2 C12(CNC(c3csc(F)c3)=O)CC(CO1)N(C(c1nccc(C(F)(F)F)n1)=O)C2 Cc1cc(F)cnc1C(=O)NCCOCCC(N1CCC(O)(CO)C1)=O Cc1cnc(C(N2CC(NC(c3ccc(-c4nnc(S)o4)cc3)=O)C2)=O)cn1 c1(C(=O)OC)ncccc1NC(c1cc(NCc2cccc(OC)c2)cn1C)=O CCC1=C(C(=O)NC(C)C(C)NC(=O)Cc2ccc(O)cc2)CCCO1 c1(C(N2CCN(C(CCOCC)=O)CC2)=O)ccc(C#N)cc1F c1(C(=O)NC(C(=O)NCCS(CC)=O)C(C)C)ccc2[nH]ccc2n1 c1(C(c2n(CCC)nnn2)NC(c2ccnn2CC)C)nc(Br)ccc1C C1(CC(=O)NC2(CN(C(=O)Cc3cccn3C)C)CC2)CCCC(=O)C1 O(NC(=O)C1=C(F)CN(C(c2cccc3ccoc23)=O)CC1)C(CC)C C1(C(C)NC(CCNC(CCCOC)=O)=O)CN(C)CCO1 C1(NC(C=CCN(CC#C)C)=O)CC2(CCN(C(c3c[nH]cc3Br)=O)CC2)C1 C1(NC(C#C)CC(C)C)CCC2(CCCNC2)C1 Cc1cnccc1C(N1CCC(C(C)NC(=O)C=CCF)C1)=O c1(CC)onc(C(N2CCC(C(N3CCC(CF)C3)=O)CC2)=O)c1C c1(C(N(CCCNC(C2(C)C(C)(C)C2)=O)CC2CCCC2)=O)cncc(F)n1 c1(SC)ncc(CC(=O)NCC2C=CC(NC(=O)CC3C=CCC3)C2)c(O)n1 CCCC(C(=O)NCC1CC(NC(=O)C(=O)NCC(F)(F)F)C1)NC(N)=O N1(C(C2CCC(CC)O2)=O)CC2(CCN(C(c3cnc(C4CC4)[nH]3)=O)C2)C1 c1(OC)cc(OC)cc(C(=O)NC2CC3CC2N(C(c2n[nH]c(C)c2F)=O)C3)c1 CCC(C)CC(C)NC(=O)CNC(c1n[nH]c(C)n1)(C)CC C1(C(=O)NC2CCC(CCNC(=O)CN3CC4C=CC3C4)C2)CCC2(CC1)CC2 c1(C(=O)NC2CCC(NC(c3n(C)nnc3)=O)C2)cnc2c(F)cccn12 N1(C(C2CCCN(C(C(C)N(CC)CC)=O)C2)=O)C2CCC1C(CO)C2 CC12CN(C(=O)CNS(=O)(=O)c3ccccc3)CC1CN(C(C1C=CCC1)=O)C2 c1(CN(C(C2C(NC(C(CC)C)=O)CCO2)=O)C)ccccc1C c1(OC)cc(C(N2CC3CN(C(C4(C)CCCCC4)=O)C3C2)=O)ccc1C N1(C(CCN(C(CCSC)=O)C(C)C)=O)CC(=O)N(C)CC1C c1(C(=O)NC2CN(CC)C2)cccc(CNC(=O)C(c2cccnc2)O)c1 C1(CC)CN(C(C2CC3(CC3)CN2C)=O)CCN1C(c1cscc1OC)=O c1(OC)ccc(C(=O)NCC2CC2NC(=O)CC2(C)CC2)c(OC)c1 C#CCCCCCC(=O)NC1(CO)CCCN(C(c2ccccc2COC)=O)C1 CS(=O)(=O)c1ccc(C(=O)NCC2CCN(C(c3ccc(F)s3)=O)CC2(F)F)[nH]1 CN1C(=O)CC(C(=O)NCCN(C(=O)C(O)CC(N)=O)C)C1c1ccnn1C C(CCCC(=O)NCC1(C(F)F)CCN(C(c2nnc(C)s2)=O)C1)SC Cn1[nH]c(=NC(=O)C2CC2NC(c2sccc2Br)=O)c2cccnc12 CCC(O)C(C)(C)C(=O)NC(C)CN(C(=O)Cc1ccc(C)nc1)C Cc1cc(C)c(NC(=O)C(c2cc[nH]n2)N(CCC(C)C)C)c(C)c1 Cc1noc(C)c1C(=O)NCC1(c2cccnc2)CCC1.C12CCC(C1)NC2=O C1(NC(C(C)SC(F)(F)F)=O)CCN(C(c2ccc(F)cc2F)=O)CC1C N1(C(C2CN(C(C)=O)C2)=O)CCC(C(=O)NC(=O)CCNc2ccc[nH]2)C(F)C1 C1(C)(CNC(=O)NCC(C2CCCO2)OC)CC2(CCC2)C1 c1(CN(C(C(=O)OCC)C)Cc2ccncc2)cc(C(F)(F)F)n[nH]1 CC1(C)CCCC(C(=O)NCCC2(C)CCN(C(=O)CCCc3cnn[nH]3)C2)C1 Cc1cnc2c(C(=O)NCC3CC34CN(C(=O)OC(C)(C)C)C4)cnn2c1 CC1CCCC1C(=O)NCc1cc[nH]c1C(=O)N(C)Cc1nc[nH]n1 C1(CC)C(=O)N(C)CCN1C(C1(NC(=O)C(C)C(=O)OC)CC(O)C1)=O C(C(C)(C)CC(=O)NC1CC(CNC(=O)CCc2ccc(F)cc2Cl)C1)OC Cc1cccc(-c2cn(CC3CCCCN3C(=O)Cc3nccn3C)nn2)n1 c1(SC)ccc(CCC(=O)NCC2CC(O)(CNC(=O)C(O)CCSC)C2)cc1 C(N=c1cc(C(N2CCC(O)C2)=O)cn[nH]1)c1ccc(C#N)o1 C=CC(C)(CCOC)C(=O)NC(C1CN(C(=O)CCc2cn[nH]c2)C1)C N1(c2nnc(COC)s2)CCC(C(=O)NCCc2ccc(I)cc2)C(CO)CC1 Cc1ccc(CNC)cc1.C12(C(N3CC(OCCNC(CS)=O)C3)=O)CC(F)C1C2 C1(N=c2nc[nH]n3ccc(Br)c23)(C(=O)NC2CCCN(C(C)=O)C2)CC1 c1(OC)ccc(C)c(CNC(=O)C(=O)NC2CC(n3cnnc3C)C2)n1 CC(C)CC(C(=O)Nc1cc(SCN2CCCCC2=O)cc(O)c1)ONC(=O)C1CC1 c1(C(N2CCCC(C)C2CCNC(C2(F)CC2)=O)=O)cccc2c1COCCN2 N1(C(CCC)=O)CCC(C(=O)Nc2cc(OC)ccc2O)C(C)C1 C1(NC(c2nocc2Br)=O)CN(C(=O)CCn2cnnn2)CC12CC2 Cc1nn(C)c(Cl)c1C(=O)NCC(C1CCN(C(=O)C(C)c2ncco2)C1)(C)C c1(C(N2CC(C(C)NC(Cc3scc(C)c3)=O)C2)=O)cnc2cccnc2c1 O=S(=O)(c1cccc(N2CCN(C3CCC3)CC2)n1)NCc1ccnc(Br)c1 C1(NC(=O)COCC2CC2)CC12CC(NC(c1n[nH]c(C3CC3)c1Cl)=O)C2 C1(O)(C)CC2C=CC1C2.C1(C(=O)NC2CCOC2)CSCCN1C(=O)CSC C1(NC(CC2CCCC(C)C2)=O)CN(c2ccnc(C#N)n2)CCC1C N1(C(CC)=O)CCCC(C(N2CCC(N(C(=O)CCc3nc[nH]n3)C)C2)=O)C1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(C)(NC(C2C(C(=O)OC)CC2)=O)CC1 c1(C(N(CCc2cn(C(C)C(=O)O)nn2)C)=O)ccc(Br)c2cn[nH]c12 c1(C(N(C2CN(C(=O)COCC(F)F)CC2(C)C)C)=O)cc2cnccc2o1 N1(C(CC2(CC)CCC2)=O)CC2CC(NC(c3cn(CC)nn3)=O)C1C2 c1(C(N2CCC(CC(=O)NOCC(F)(F)F)CC2)=O)ccn2ccccc12 Cc1cc(NC(C2CCN(C(c3ocnc3C)=O)C23CC3)=O)ncc1F C(CCN(C(=O)CC(C)(C)O)CCOC)(C(C)C)NC(CCN(C(CC)CC)C)=O C=CC1COCC1NC(=O)C(CCOCCO)NC(=O)CCc1ccccn1 C#CCCCC(C)C(=O)NCC1CC(C)(C)CN1C(c1ccnc(S)c1)=O N#Cc1cc(S(=O)(=O)N2CCC(C(=O)Nc3cnccn3)C2)ccc1Br C1(C(=O)NCCOCCC(=O)NCC(C)(C)n2cccn2)CCCCO1 CC(C)CC(C(=O)NC(C1CC=CCC1)C(=O)NCC(C)(C)CCCO)C(N)=O c1(C(N2CC(O)(C(C)NC(=O)CNC(N)=O)C2)=O)ncc[nH]c1=O C(CCCC)(C(=O)Nc1cnn(C)c1C#N)NC(CN(CCC)C)=O c1(C(=O)NC23C(CN(C(C(CC)C)=O)C2)C3)cc2[nH]nc(C)c2cn1 CCC(CC(=O)N(CC(C)C(=O)N(C)Cc1cccc(O)c1)C)SC c1(CN2CC3(CC(C(=O)Nc4c(C)ccc(F)c4)C3)C2)cnc2cccnn12 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)CN3CCCC3C)C2)sc1S(N)(=O)=O CCC(C)(C)CCCC(=O)N1CCC(N(C)C(c2cnn(CC(F)(F)F)c2)=O)C1 c1(C(N(C2CN(C(=O)Cc3cnoc3)CC2(C)C)C)=O)cc2c(=O)[nH]ccn2c1 c1(C(=O)NCCC2(NC(C3(N4CCOCC4)CC3)=O)CC2)ccc2ncnn2c1 N=c1ncc(C(=O)NC2CC(OCC(=O)NC3CCOC(CCN(C)C)C3)C2)c[nH]1 c1(CC(=O)NC(CNC(CC(C)c2cnn(C)c2)=O)C2CC2)ccc(Cl)nc1 c1(CNC(N(C2(C(=O)NCC(COC)CO)CCOCC2)C)=O)ccc(F)c(F)c1 C1(NC(CCCn2c(C)ncc2)=O)CC2(C1)CN(C(c1ccccc1CO)=O)C2 c12cc(c(OC(F)F)cc1Br)NC2=O.N1(C(=O)OC(C)(C)C)C(C(=O)O)CC2CC12 c1(CC(=O)NC(COCCOC)Cc2ccccc2)ccc(OC(C)C)cc1 c1(OC)ccc(CCCC(=O)NC2CCCN(C(=O)Cn3ccnc3C)C2)cc1 c1(OC)ccc2c(c1)C(NC(=O)CCCN(C)C)CCN2 c1(N)ccc(C2(NC(=O)NC)CCC2)cc1.C(=O)(CCCC1CC1)C(C1C(NC)C1)=O C(C(CC)(CC)CO)NC(c1cc(Br)c(Cl)s1)c1n(CC(=C)C)nnn1 CCC(CC)CCC(=O)N1CCC(C(=O)NC2CCCN(CC)C2)C(O)C1 c1(NC(C2(C(N(C(C)C)C)=O)CCC2)=O)ccc(N2CCCCCC2)cc1 c1(-c2cccc(OCCC)c2F)c[nH]c2cc(C(=O)NCCCCCO)ccc12 C1(NC(=O)CC2CC2)CN(C(=O)CCCn2ccnc2)CC1O.N1(C)CSCC1=O c1(CCC(=O)NC2CCC(CNC(CC(=O)OCC)=O)CC2)ccc(F)c(Br)c1 N1(C(CCC(C)(C)C)=O)CCC2(CCC(NC(=O)CC3CC(F)C3)C2)C1 C1(C)(C(=O)OC)CC(F)CN1C(=O)C(Cc1ccccc1Br)CC CN1CCN(C(=O)CCC2CCCC2)CC1C(=O)NC1C=CCCCC1 C(C(C)CN=c1[nH]c2ccc(Cl)cc2s1)NC(c1cnc(C(C)C)[nH]1)=O c1(OC)ccc(C)nc1C(C(=O)CC(C)C(F)F)=O.C(C(C)(C1CC1)SC)N c1(CCC)cc(C(=O)NCC2(CNC(C)=O)CC23CCC3)cc(O)n1 n1(CC(=C)C)nnnc1C(c1cc(C2CCC2)[nH]n1)N(C(c1ccno1)C)CC C(CCCC(CO)NC(c1ccnn1C1CCOCC1)=O)NC(=O)C=C1CCC1 N1(C(=O)Nc2c(SC)cc(F)cc2)CC2CC(C1)CS(=O)C2 Cc1nc(C)c(CNC(C2(C)CCN(C(C3CC(O)C3)=O)C2)=O)[nH]1 c1(N2C(C)C(NC(=O)CCc3ccoc3)CC2)nc(=NCC2CC2)[nH]c(Cl)n1 CC1C(C(=O)N2CCCC2C(N2CCCC(CO)C2)=O)=NOC1C N1(C(C(CC)OCC)=O)CC(NC(c2scc(C)c2Cl)=O)CCC1C n1(CC)cc(Br)c(C(N2CCN(CCCSC)CC2)C(=O)Nc2cccs2)n1 C1(NC(C(CSC)N(C)C)=O)CCCCC1NC(=O)COCC(n1cncn1)C c1(C(=O)NCCC2CCCN(C(c3c(C)nccc3)=O)C2)nccc(Cl)c1F C1(C(C)(C)NC(C2CCCN2CC(F)(F)F)=O)CN(CCO)CCO1 c1(CS(=O)(=O)Nc2c(OC(C)C)cccc2)cc(Cl)c(Br)c(Cl)c1 N1(C(C=CC)=O)CC2(C1)CN(C(c1csc(CC(C)C)n1)=O)C2 CN(OCC(F)(F)F)C(=O)C(CNC(c1ncc(F)cc1F)=O)CC1CC1 c1(C(N(C(C)CCNC(C2CC(CCF)C2)=O)C)=O)ccc2c(c1)C(=O)NCC2 C1(C)(NC(C(c2cc(C)sc2)(F)F)=O)CCN(C(C2(C)CC2C)=O)CC1 CCCCC(CC)C(=O)NCCCNC(c1cc(N2CCNC(=O)C2)ccn1)=O CC1(C)CN(C(c2csc(C#N)c2)=O)CC1NC(c1cc(C(F)(F)F)c[nH]1)=O CC(=O)CCCC(=O)N(CCCNC(=O)CC1CCC(C)(C)CO1)CCO C1(C(=O)NCC(CC)NC(c2cccc(CCO)c2)=O)(CO)CC(F)(F)C1 C1(N)CCCCN(C)C1=O.C(CC(C(=O)NCC1CCCCC1)NC=O)SC n1(CC(CC)O)cc(CN(C(=O)Cc2nc(-c3cccnc3)cs2)C2CC2)nn1 C1(C#N)(c2cn(CF)nn2)CC2CC2C1.N12CCCC(C1)C2.C12CC1(F)C2.C(=O)OC c1(CC(N2C(CNC(c3cn(CC)nn3)CC)CCC2)=O)cnn(C)c1C C1(NCC)CC(CF)C1.C(C(C)N(CC=O)CC)OCC C1(CCNC(C(CC=C)CC=C)=O)CC(N=c2[nH]c(Cl)ncc2C(C)=O)C1 N1(C(C2(C=C)CCC2)=O)CC(CNC(c2sccc2OC)=O)N2CCC1C2 c1(C(NOCCOCC#C)=O)cccnc1CNC(c1scnc1CC)=O c1(C(COCCn2cncn2)NC(N(C(C)C)CC)=O)ccc(Cl)cc1 N1(C(CCCC(CC)CC)=O)CCC2C(CCCN2C(C)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CC(C(Cn2cc(CCN(C)C)nn2)F)C1 C12(C(=O)NCCCOC3CCN(C(C4(F)C(C)C4)=O)CC3)CCCN1CCC2 C(C)(C(C)(C)C(=O)N(C(C)CN(C)C)C)NC(COCC(=O)NC)=O C1(CNC(c2c(C)nc(CC)o2)=O)CC2CCC1N(C(C1CCC3CC13)=O)C2 C=CC1CN(C(=O)C(F)(F)c2cnn(C)c2)CC1NC(c1cccs1)=O Cc1cc(N)c(C(N2CC(C3CN(C(=O)C(C)N(C)C)C3)C2)=O)c(F)c1 C1(C(=O)NCC(C#C)CC2CC2)CN(C)CCN1C(=O)CC(C)(C)CN(C)C c1(CC(N2CC(C(C)NC(C(CCC)OC)=O)C2)=O)c(Cl)ccc(O)c1Cl C1(C2(C)N=N2)COCCN1C(C1CC1CNC(=O)CCCN1CCOC1=O)=O C(=O)(C(F)CC(C)(C)NC(=O)NC(c1cc(F)ccc1OC)C)OC Cc1ccc(C(C2CC2)NC(C2CCN(C(=O)C(Cl)Cl)C2)=O)cn1 c12ccc(cc1)C(=O)NCC2.C(C1=NOCC1)CNC(N)=O C(=O)(CCCCC(C)(C)C)NCC(CC)(C)NC(c1ncn2ccccc12)=O c1(CN2CC(F)CC(C(N3CCn4nccc43)=O)C2)ccc2ncnn2c1 Cc1ccccc1C1CCCN1C(=O)NCc1ccccc1OCc1ccco1 C(=O)(C1=CCCOC1)N1C(C(=O)NCC(=C)F)CC1C C1(C(N2C3C(C(=O)OC)C(C3)C2)=O)CN(C(=O)C2CC2)CC(C)O1 C1(CNC(=O)CSC2CCOC2=O)COCCN1C(=O)Cn1cccc1 C1(CNC(C(C)C(F)F)=O)CC(F)(F)CN1C(=O)COCc1ncnn1C N1(C(c2cccnc2S)=O)CC2(CCN2C(C2CC3C=CC2C3)=O)C1 c1(OC)coc(C(N2CCCC(CN(C(=O)C3=CCCOC3)C)C2)=O)cc1=O Cc1cnc(C(N2CCC(NC(=O)CC3CCCC(C)O3)C2)=O)cc1C#N N1(C(CCC(=O)OC(C)(C)C)=O)CCCCC2C(OC(c3ccoc3)=O)C12 CN1CCCC(F)(C(=O)NCC2CN(C(=O)Cc3csc(=N)[nH]3)CCO2)C1 c1(Cc2cc(C(=O)NCCNC(C3CC(COC)C3)=O)on2)cccc(Cl)c1 N1(C(C(C)c2ccco2)=O)CC(NC(=O)Cc2cncn2C)CC1C Cc1cccc(OCCNC(=O)CN2CCOCC2c2ccc(C(=O)O)o2)c1 c1(C(N(C)CC2(NC(C3C(C)CCC3)=O)CC2)=O)ccnc(OC2CC2)c1 Nc1c(C(=O)NC2CC2NC(=O)C(c2ccccc2F)(F)F)cnn1CCO CC1OC2(C(N3CCCN(C(C4CCCC4)=O)CCC3)=O)CCC1CC2 C1(NC(C(=O)NC2CCCC2n2cccn2)=O)CCCCCC1 Cc1cc(Cl)c(S(=O)(=O)N2CCC(NC(=O)OC(C)(C)C)C2C)c(Br)c1 C1(NC(CCC=C(C)C)=O)(CNC(=O)C(n2ccnc2C)C)CC2CCC1CC2 c1(C(N2CC(N(C)C(c3cnc[nH]3)=O)C(C)(C)C2)=O)ccc2nnnn2c1 N1(Cc2csc3ccc(C)cc32)CCC(C2CCCOC2)CC1 c1(C(C)C2CC2)nc(-c2ccccc2Br)nn1C1CCS(=O)(=O)C1 N1(C(C(=O)OC)C)CCN(C(C23CC(CCN(C)C)(C2)C3)=O)CC1 CC(C)C(C)(C)C(=O)NCC(C1CCCN(C(c2ccc(F)o2)=O)C1)(C)O C(N=c1nc(C2CCOCC2)[nH]s1)C1CCC(C(=O)C=Cc2ccncn2)CC1 Cc1cc2[nH]c(C(=O)NC3CN(C(=O)CCOc4cccnc4)CC3C)cc2s1 CCS(=O)(=O)c1ccc(C(N2CCCC2CN(C(=O)C2=CCCS2)C)=O)cc1C C(C(F)(F)CC(O)CO)N(C(c1cc(SC)nn1C)C(=O)NCC=C)C C1(NC(c2c(C)noc2)=O)CC2(C1)CN(C(=O)CS(=O)(=O)Nc1ccccc1)C2 c1(C(C)NC(C(CC)(CC)CO)=O)ccc2c(c1)CN(C(c1cnc(Cl)s1)=O)C2 c1(OC)cc(C(N2CCCN(C(C3CC4(CC4)C3)=O)CC2)=O)cc(Cl)n1 N1(C(c2c(N)ccc(C)c2)=O)CC2CCC(NC(C3CC(CF)C3)=O)CC2C1 C1(CNC(C(C)C(F)(F)F)=O)CN(C(c2cc(Cl)no2)=O)CCC1(F)F C12(COC)COC(C(=O)NC(C3CN(C(c4cccs4)=O)CCO3)C)(C1)C2 C(=O)(CC(C)(C(F)F)N(C)C)NCc1nc(CNC(C(CSC)C)=O)nc(O)c1 Cc1cc(C(N2CC(C3(NC(C4CC4Cl)=O)CC3)C2)=O)ccc1C(C)C c1(C(=O)NC2C(NC(C=CCC)=O)CS(=O)(=O)C2)cnc2c(c1)nc(O)n2C N1(C(c2cc(C(C)=O)oc2)=O)CC2(COC(CNC(=O)CC(O)C(C)C)C2)C1 N1(C(c2c[nH]nc2C2CC2)=O)Cc2[nH]nc(C(N3CCc4ccncc43)=O)c2C1 c1(CC(N2C(CN(C(=O)CC3CC3(Cl)Cl)C)CCC2)=O)ccnc(Cl)c1F C(=O)(C(C)(C)C(=O)N1C(C(=O)NC2(C3CC3)CCOC2)CC1C)OCC C=CC(C)CCN=c1ccc(S(=O)(=O)N2CC3CC(C2)C3(C)C)c[nH]1 C1(C(=O)NCCSCC(C2CCOC2)NC(=O)Cn2cncn2)C=CC=CC=C1 C#Cc1ccc(CC(=O)NCC(C(=O)NCCC2CC(CF)C2)N(C)C)cc1 N1(C(C(CC)C)=O)CC(NC(=O)C(C)OCC(=O)NC(C)(C)C)CC(F)C1 CN1C(=O)CN=C1NC(=O)NC1CC2CCC(C1)N2C C1(CCOC)(NC(=O)CC2CCCO2)CCN(C(C2CCCO2)=O)CC1 CC(C)(C)C(C#N)C(=O)NCCC1CCCN(C(c2cc(Br)cnc2)=O)C1 CC1CC(NC(=O)CSC(F)(F)F)CCN1C(=O)CCN1CCC(F)C1 C(CCC(=O)NC1CC(NC(=O)COC(C)CCc2nccs2)C1)N(C(C)=O)C C1(C)(C(=O)NCCC(CNC(c2c(CC)cccc2)=O)O)CC(C(C)C)=NO1 c1(C(=O)NCC(C)NC(c2cnc(NCC)c(Cl)c2)=O)cccn2cnnc12 c1(C(=O)NCCNC(C(C)(C)SC)=O)cc2c(C)c(Br)ccc2[nH]1 C(=O)(CC(C)C(F)F)NC(C)C(C)NC(=O)CCc1nccs1 C1(NC(CC=C)=O)CCC12CCN(C(C13C4C5C1C1C3C4C51OC)=O)CC2 C(=O)(CCCCN=[N+]=[N-])NC(C(C)C)CNC(c1cncs1)=O C(c1ccc(Cl)c(COC(=O)Cc2ccc(Cl)cc2F)c1)=CCCC c1(OCC(CN2C(NC(=O)Nc3ncccc3F)CC2)O)cccc(F)c1 C#CCCCCCCC(=O)N1CCN(C(=O)C(C)Cc2cccnc2)CC(O)C1 C1(C(=O)OC)CCCN1C(=O)CCc1ccc(N(C)C(C)C)[nH]1 CC1(C)C(C(N2CC(CNC(c3ccoc3Cl)=O)C(C(F)(F)F)C2)=O)C1(C)C c1(CC)nccnc1C(=O)NCC(C)(CNC(=O)Cn1ccnn1)OC c1(C(N2CCCCC2CCO)=O)cc(OC(F)(F)F)ccc1O N1(C(c2c(C)cncc2)=O)CC(C)(C)CC1CNC(c1cnc(C(F)(F)F)s1)=O C1(NC(C(=C)C(F)(F)F)=O)CN(C(=O)CN2CCOC2=O)C2(CCOC2)C1 N1(C(=O)NCCOC(C)C)CCC2C(CCCN2C(C)=O)C1.c1(N)ccc(OC)cc1 C1(C(=O)NCc2nc(Cc3ccccc3)no2)(OC)CCN(C(C)CCO)CC1 c1(CC)nc(N(C)C)[nH]c(=NCC2(P(C)(C)=O)CC2)n1 CC1CN(C(=O)CCNC(N)=O)CC1CNC(c1cccc(C2(C)CCC2)c1)=O C=CCC(CNC(=O)C=CCC1(NC(C2CC=CC2)=O)CCC1)CC(C)C CCC(C(=O)NCC1(O)CN(C(C2C3CCC(C3)C2C)=O)C1)C(F)(F)F C1(CCC)CN(C(c2cn(C)nc2C)=O)CC1NC(C1(OC(C)C)CCOC1)=O C(=O)(C(C(C)C)NC(=O)CCn1cccc1)N(C)CC N1(C(C=CCC)=O)CCC(C)(C)C(C(=O)N(C(CCCC)C(C)C)C(C)C)C1 N1(C(C(CCC)(C)O)=O)CCN(C(=O)C(CC)(CC)CO)CC12CC2 N1(C(CC=C)=O)CCC(C(N2CC(CO)C(C)(C)C2)=O)C12CCC2 CC1(C)CN(C(=O)C#CC2CC2)CCC1NC(=O)CCCNC(N)=O Cc1csc(=O)n1CCN(CC(=O)NCCCCl)CCc1ccccc1 N1(C(C2CC=C(C)CC2)=O)C2CC1CN(C(c1ccncc1Br)=O)C2 C(=O)(C(CO)C(C)(C)C)NC1(C(=O)NCC2(OC)CC(C)(C)C2)CCSC1 N1(CCNC(c2cn(C3CCN(C(C(C)OC)=O)C3)nn2)=O)CCNC(=O)C1 C(=O)(C(F)C(C)(C)O)N1CC(O)(C(C)NC(=O)CCc2ccc(N(C)C)nc2)C1 C(C(N=[N+]=[N-])C(=O)NC(C)(CC)CCNC(c1ccc(C)nc1C)=O)OCC N1(C(CC2(COC)CC2)=O)CCCCCC1CNC(=O)C=Cc1ccc(C)nc1 c1(NC2CCCC(C(F)(F)F)C2)[nH]c(=NCc2ccns2)nc2scnc12 N1(C(C2ON=C(C)C2)=O)CCN(C(=O)Cc2ccc(F)cc2C)C2COCC12 Cc1nccc(C(N2CCN(CCNC(C3(CCC(F)(F)F)CCC3)=O)CC2)=O)n1 c1(C(N2CCN(C(C3(OC)CC(C)C3)=O)CC2C)=O)cc2ccccn2c1 c1(NCCCCC(C)NC(C23CCC(C)(C2)OC3)=O)c([N+](=O)[O-])cnn1C N(C(=NCCCF)NCC1COC(C)(C)C1)CC1(COC)CC=CC1 C1(n2c(C(c3ccc(-c4cc[nH]n4)s3)F)nnn2)CCC2(CC2)C1 C(=O)(C1CCOc2ccc(F)cc21)N(C1CCN(C(c2coc(Cl)n2)=O)CC1)C N1(C(C=C(CNC(CN2CC(C)(OC)C2)=O)C)=O)CCOC(C)(C2CC2)C1 c1(C(N(CCCCNC(CC(C)(C)OC)=O)C)=O)cccn(C)c1=O N1(C(C2C(OC)C2)=O)CCC2(CCC2NC(C23CCC(=O)N2CCS3)=O)CC1 C(C(CC(=O)NC1C2CCCOC12)NC(=O)CCc1cn(C)cn1)OC C1(C(F)F)(N(C(c2ccc(C)cc2)=O)CCc2ccccn2)CC2CCC1CC2 CC(C)(C(=O)NCCCOCCNC(=O)C=CCO)c1cc[nH]n1 c1(OC)nccnc1C(N1CCN(CC(=O)NCCc2ccc(C)cc2)CC1)=O C1(C(N2CCN(CCC#C)CC2)=O)CCN(C(=O)C(C)C)C12CCC2 N1(C(c2nccc(C)n2)=O)CCCC(NC(c2cc(C)oc2C)=O)CC1 c1(-n2cc(C(=O)NCC(=O)O)nn2)cc(F)cc(F)c1 c1(OC)ccc(NC(=O)CC(C)n2ccnc2)cc1F.C1C(O)CC(=O)N1C Cc1ccc(C(=O)NC2CCCC(C(=O)NC(=O)C3CC3)C2)nc1 N1(C(C(n2ncc(C)c2)C)=O)CCC(C(=O)NCc2cnco2)CC1(C)C CC1(C)CCN(C(c2cc(CCO)on2)=O)CC1CNC(=O)CC1CCOC1 C1(O)(CC(C)C)CCN(C(=O)C(C)N(C(c2coc(C(F)F)c2)=O)C2CC2)C1 n1(CC)cc(C(N2CCC2(C)CC(=O)NCC2(C)CC2(F)F)=O)c(C)n1 c1(CNC(C2C(CC)C2)=O)ncccc1CNC(=O)CCCNS(C)(=O)=O c1(N2CCCCC(CNC(C3N(CC)CC3)=O)C2)c(F)cc(C#N)cc1[N+](=O)[O-] C1(C)(C(=O)NCC(=C)C)CN(C(c2cnc(O)n2CC)=O)C(C)(C)C1 C1(CNC(c2cc(-c3ccncc3)no2)=O)CCN(C(=O)Cc2cn[nH]c2)C1 C1(CC(=O)N(CCCCN(C(C2(CC(C)=O)CCC2)=O)C)C)CS(=O)(=O)C1 C(=O)(C(C)CCCC(C)=O)NC(CCC#C)C(=O)NC(c1cccnc1)C C1(C(N2CC(C=C)C2C(N2CC(OC)C(O)C2)=O)=O)CCC2(CCC2)O1 C(=O)(CCCCC(=O)NC(CCC1CCC1)C(=O)NC1C=CCC1)OC c1(NC(C2(C)CCN(C(c3c(CC)csc3)=O)C2)=O)cccc(CO)c1C c1(C(N2CC(C)C(NC(C3CC(=O)N(C)C3)=O)C2)=O)ccc(F)c2ncccc12 Cn1cc(C(=O)NCCCCNC(N)=O)c(O)n1 C#CCC(O)C(=O)N1CC(NC(c2cc(C)n(C(C)C)n2)=O)C(C(F)F)C1 C=CC(C)(CCOC)C(=O)NCCCN(C)C(C1CCc2nccn2C1)=O C1(C(=O)NCC(=C)CCNC(c2ccc(=NC)[nH]c2)=O)CC2CCC(C1)C2(F)F CCC(C)C(=O)NCC(=O)NCCN(C(c1cc(CO)on1)=O)CC C(=O)(C(F)(F)C(F)(F)F)NCC1CC(CNC(=O)CC(=O)NCC2CCC2)OC1 c1(C(N2CCOCC(NC(CCC)=O)C2)=O)ccc2c(c1F)CCC2 CC(C)(C)CC(C)(C)C(=O)NC1CC2CC1N(C(C1CCCO1)=O)C2 N1(C(CCc2onc(SCC)n2)=O)CCOC(C(NCP(C)(=O)OCC)=O)CC1 c1(NC(c2c(C)cccn2)=O)cc(F)c(-c2cn(CC3CCOC3)nn2)c(F)c1 c1(C(=O)NCC(C(=O)NC2(C)CC=CC2)O)cc2ccncc2[nH]1 C=CCCCCC(=O)NC1CC(CNC(C2COCCC2(F)F)=O)C1(C)C c1(C(N2CCN(C(CCC(=C)C)=O)CC2CC)=O)cc(Br)c(C)cc1F c1(C(N2CCC(CCC(=O)N(CCC)CCC)C2)=O)cc(C)n(C)n1 C1(NC(COCCC)=O)CC2CCC1CN(C(=O)Cc1ccc(OC(C)=O)cn1)C2 CCS(=O)(=O)CCNC(=O)CC1CCC(NC(=O)C(C)OCCC(C)C)C1 N1(C(C(=O)NCC(CC=C)NC(c2cnc(O)c(F)c2)=O)C)CCP(C)(=O)CC1 C(=O)(CC(F)(F)C(F)(F)F)N1CC(O)(CCNC(c2scc(C#N)c2)=O)C1 N#Cc1cc(COC(=O)CCc2ccc(Cl)c(F)c2)ccc1O C1(C(N(C)CC2CN(C(=O)C(F)C3CCCC3)C2)=O)CCC(C)(C)O1 c1(N2C3CN(c4ccnc(SC)n4)CC32)ncnc2[nH]cc(I)c12 Cc1ccc(C(=O)NC2CCN(C(=O)C=Cc3cn[nH]c3)C(C)C2)c(O)c1C C1(N(C(=O)COC2(C)CCC2)CCC)CCN(C(c2cnccn2)=O)CC1 c1(C(=O)NC(C)C(C(C)C)N)ccc([N+](=O)[O-])s1.C(CCCC=O)OCC CC1(CO)CCCN(C(C2CC3(CCCO3)C2)C(=O)NC2CCC2)C1 C(=O)(C(C)(C)C(C)(C)C)N1CCC(CNC(c2c(CC)occ2)=O)(OC)CC1 C1(NC(C(CC)N(C)C)=O)CCN(C(c2cc(C(N)=O)co2)=O)CC(C)(C)C1 CCC(CC(=O)NC1(CNC(=O)Cc2nocc2C)CCCC1)c1ccccc1 N1(C(C)C)CCC(C(=O)N(CCCNC(C2CCC(C)C2)=O)C2CC2)CC1 c1(C(=O)NCC(C)NC(c2cnc(C3CC3)[nH]2)=O)cnn(-c2ccncc2)c1 C=CC(C)(O)CC(=O)N1CC(NC(=O)Cc2ccc(O)c(OC)c2)CCC1C CC12COCC1(C)CN(C(=O)NC1C3C(=O)OCC13Br)C2 c1(NS(C)(=O)=O)cccc(S(=O)(=O)NCC2(O)CCOC2)c1 N1(C(c2ccn3ccnc3c2)=O)CC2CCCN(C(c3ccnc(Cl)c3)=O)C2C1 C1(C(=O)NCCN(C(c2cc(C(=O)OCC)n[nH]2)=O)C)CC2(CCC2OC)C1 c1(C(N(CCNC(=O)Cn2cnnn2)CC)=O)cc2c(O)ccc(F)c2[nH]1 C(=O)(C1=CS(=O)(=O)CCC1)NC(CCCC)CNC(=O)CCc1cnco1 C1(N(C(c2cn3cccc(C)c3n2)=O)C)Cc2ccccc2C1O CCC1CCN(C(CN(OC)CC(N)=O)=O)c2cc([N+](=O)[O-])ccc21.OC N1(C(C=CSC)=O)CCC(N=c2[nH]c3ccccc3o2)CC1C C1(C(N(C(C)CNC(=O)CCOCC(F)(F)F)C)=O)CC2(CCCCC2)C1 N1(C(C(CNC(c2c(C)csc2)=O)CC2CCCC2)=O)CC2(CCC2)CC1C c1(CCC(=O)NC2C(CNC(c3[nH]cc(C#N)c3)=O)C2)c[nH]c2ccccc12 c1(NC(C(c2cc(C)c(Br)cc2)C)=O)nc2c(s1)COCC2 C(=O)(C(O)CSC)N(CC(C)NC(=O)CCN(C)C(C)=O)CC Cc1ccc2occ(C(N3CC(NC(c4cnncc4C)=O)CC(O)C3)=O)c2c1 c1(CN2C(c3cnn(CC)c3)C(=O)NCC2)scnc1C.CCC(=O)OC c1(OC)cc(C(F)(F)F)ccc1CNC(C1CC(Nc2ccc(Cl)cc2OC)C1)=O N1(C(C2(CCNC(=O)C=CC(=O)NC(C)C)COC2)=O)CCC(CO)CC1.COC c1(C(=O)NC(C2CCN(C(c3c(C)ccc(F)c3)=O)C2)C)n[nH]c2c1COCC2 C1(CNC(c2cccc(CC)n2)=O)CN(C(c2ccc(N(C)C)s2)=O)CCC1C C1(C(N2CC(O)(CNC(C34CCC(CC3(F)F)C4)=O)C2)=O)CC2(CCCC2)CO1 CC1=C(C(=O)N2Cc3ccccc3CC2C(F)F)C(C)(C)CCC1 C1(NC(C2CCN(C(C)=O)C2)=O)CC12CCN(C(c1cc(C#N)[nH]c1C)=O)CC2 CC(C)(C)C(CNC(c1cc(C2CCOCC2)on1)=O)NC(C1(O)CCOC1)=O C1(N(C(CCC=CC)=O)CC)CCCN(C(=O)CC2CC(C)(C)CCO2)CC1 C1(C(N(CCCOCCNC(COCCCC#C)=O)C)=O)CNC(=O)N1 C1(CNC(c2cnc(OCC)nc2)=O)C2CCCC1N(C(=O)C(C)CCSC)C2 C1(C)(CC)C=C(C(=O)NCCC(C)(C)C(=O)N(C(C)CCSC)C)C1 Cc1nc(N2CC(C(C)NC(c3cnnc(O)c3)=O)C2)cc2nncn12 CC(CCNC(=O)CN(C)C(=O)OC(C)(C)C)NC(=O)CSC(F)(F)F c1(C(N(CCNC(CCN(C)CC)=O)C(C)C)=O)cncc2n[nH]cc12 C1(C)(C(=O)NCC(C)CN(C(=O)CSCc2cccs2)C)C=CCCC1 CCC(C(=O)N(CCCNC(c1cscc1F)=O)C(C)C)OC1CCCCC1 C(=O)(C(C)(COC)COC)NCC(C(=O)NC(CCOC)C(N)=O)O CCCC(O)CC(=O)NC(CNC(c1ccc(OCCF)cn1)=O)C(C)C c1(C(N2C(C)(CNC(c3ccn(CC)n3)=O)CC2)=O)ccc(-n2ccnc2)cn1 N1(C(c2ccc(CC)s2)=O)CCN(C(=O)C2=C(Cl)CCC2)C2CCCCC2C1 C#Cc1ccc(C(=O)NCC2CC(CNC(=O)CCNS(=O)(=O)CC)CO2)cn1 c1(C(N(CCCNC(C2CC=CCO2)=O)C(C)C)=O)cc(O)nc(O)c1 C(=O)(C1=CCCCCC1)NC1CN(C(C=Cc2n(CC)ncc2)=O)CC1F C1(C(=O)NCCc2cnsc2)CCCCC1NC(C1(CCF)CC1)=O C(=O)(CCC(C)S(C)(=O)=O)N1CCC(C2CC2)(CNC(c2c(C)ncs2)=O)C1 c1(C2CC(C(N3CCC(NC(C4CC4C(F)(F)F)=O)C3)=O)C2)cccc(Cl)c1 Cc1ccc(N)cc1C(N1C2CCC1C(NC(c1ccn(CCO)c1C)=O)C2)=O C1(CNC(c2cnc(O)o2)=O)CN(C(c2cccc(C3CCC3)c2)=O)CCCO1 c1(C(N2CCC(C)C(NC(=O)CCF)C2)=O)ccc(F)c2occc12 c1(C(=O)NC2CN(C(C3C(CC)CCCC3)=O)C(C)C2)cnc(Cl)cc1Cl C1C(CC(C)C)C(=O)N1.C(C)(CC)(CC(=O)OC)NC(C=CC)=O C1(C(C)NC(C2CC3CCCC23)=O)CCN(C(C2SCCS2)=O)CC1 Cc1nsc(C)c1C(N1CC(C(O)C(N2CCOC(C(N)=O)C2)=O)C1)=O c1(C(C)(C)C(=O)NC2CC2N(C(c2csc([N+](=O)[O-])c2)=O)C2CC2)ccc(F)cc1F c1(CCC)ccc(N)c(C(=O)NCC(C)N(C(=O)CSc2nncn2C)C)c1 c1(C(N2CCC2)=O)ncccc1N.C12CC(C1)NC(=O)CO2.C#CCS N1(C(C(F)OC)=O)CCCCC(NC(c2ccncc2O)=O)C1 N1(C(=O)Nc2cccnc2)CCC2(CC1)CC2Br N1(C(C2N(C(C)=O)CCC2)=O)CC2CCC(C1)N2C(c1cncc(C)c1Cl)=O CCCC(C)CC(=O)N1CCCC(C)(NC(=O)CCn2cccn2)C1 C(=O)(C1CCSc2ccccc21)NCc1scc(CNC(c2c(C)noc2)=O)n1 C1(OC)CCCC(C(N2CC3CC2C3CNC(c2nn(C)cc2Cl)=O)=O)C1 C(CN=C(NCCc1cccc(SC)c1)NCC1COC(=O)N1)SC C1(NC(c2ccc(F)c(F)c2)=O)CCSC12CN(C(c1ccc(F)cn1)=O)C2 C1(N(C(=O)C2CC2)C(c2ccco2)=O)CCN(C(C2CC2Cl)=O)CC1.CC C1(CN2CCC(NC(COCCCC)=O)C2)CCC2(CCC2)O1 c1(NC(C2C3CC2N(C(c2cccnc2Cl)=O)C3)=O)ccc(I)c(F)c1 CC1C(NC(=O)CC2CSC2)CCCN1C(=O)CC1CCC1 N(C1CC(C)n2ccnc21)C(c1cn(CCNC(C(F)=CCC)=O)nc1C)=O c1(CC(=O)N(C2(C(=O)NC34CC(CO3)C4)CCC2)C2CC2)cccc(O)c1 N1(C(CC2C(C)(C)C2)=O)CCC(O)(CNC(C2CCCC(O)C2)=O)C1 N1(C(c2c(Cl)cncc2Cl)=O)CC2CC(C1)N2C(c1cnc(Br)s1)=O c1(C(C)(C)C(=O)NC2CCC2NC(c2ccc(CO)cc2)=O)cc(F)cc(F)c1 C=CC(C)CC(=O)NC(c1nocc1C(N1CCOCC1CN(C)C)=O)C C(C(=O)Nc1cncc(C(F)F)c1)(C(C)(C)C)NC(c1nccc(CC)c1)=O N1(C(C23CC(C2)C3)=O)CCc2onc(C(N3CCC4NC(=O)NC4C3)=O)c2C1 C1(=O)CC(CC)CN1.C1(C(N(C2COCC2O)CCC)=O)(N(C)C)CC1(C)C C1(C(N2CCC(N(C(=O)Cc3cccs3)CC)CC2)=O)CC(F)(F)C1(C)C N1(C(CCC(C)C)=O)CCC(C2(O)CN(C(=O)COCCOCC(F)F)C2)CC1 c1(CC)cccc(C(=O)N(C2CCCN(C(=O)CCOCCOCC)C2)C)c1F c1(OC)cccc(S(=O)(=O)CCC(=O)NC2(CO)CCC(F)(F)CC2)c1 N1(C(=O)Cc2ccc(F)cc2)CC2CC1CN2C(c1cc(Cl)cc(Br)c1)=O C1(NC(CC(C)O)=O)CN(C(c2cnc(C3CC3)nc2)=O)CC1F c1(C(=O)NC2CN(C(CCC)=O)C23CCC3)cc(C)c(Br)c(C)c1 CN1CC(CCNC(=O)COC2(C)CN(C(=O)C(O)C3CCCC3)C2)CC1=O c1(C(N2CCC(n3cc(CC4N(C)CCC4)nn3)C2)=O)cccnc1Cl C#CC1CN(C(C23CCCCC2C3C)=O)CCN1C(=O)Cn1nnnc1C C(CC(=O)NC1C2CCCOC12)(C(C)OC)NC(c1cc(CC)n(C)n1)=O C(C(C)(C)CNC(c1nn[nH]c1Cl)=O)N(C(=O)C(=O)NCC1CC1)C Cn1cc(C(=O)N(CCN=c2nc(C3CC3)[nH]s2)C2CC2)c(=O)c2cnn(C)c12 c1(C(=O)NCCCCC(C)NC(CSCC(C)C)=O)cc(F)cnc1O C1(NC(c2cc(CCC)n(C)n2)=O)CCCN(C(=O)CSC(=N)N)C1C C1(CC=C)(C(=O)NC2COC(C)C2)CCN(C(=O)COc2ccsn2)C1 Cc1ccc(-c2nc(-c3cc(C(F)(F)F)cs3)n(CC3CCCO3)n2)cc1 c1(NC(CC)Cc2cccnc2)nccc(=NCCC2CC2c2ccc(C)cc2)[nH]1 N1(C(C(CCC)(C)O)=O)CC2CCC1CN2C(C12CCCC1C2(F)F)=O C(=O)(CCC(N)=O)NC1(C(=O)NC(c2ccns2)C)CC1(C)C c1(CC(N2CC(O)(CNC(=O)CSc3n[nH]c(O)n3)C2)=O)sc(O)nc1O CCC(C)C(CC(=O)NC1CC(C)(C)C1)NC(C1(C)CC=CC1)=O C=CC(C)CC(=O)N1CCC(C(N2CCC(N3CCCC3)C2)=O)C1 c1(C(=O)NC2CCC(NC(CCCN(C)C)=O)CC2)cc(Cl)c2[nH]c(O)nc2c1 N1(C(CC(CNC(C2(C=C)CCCC2)=O)OC)=O)CC(O)CC(O)C1 C1(NC(C(C2CC2)OC)=O)CN(C(c2coc(-c3csc(C)n3)c2)=O)CCC1O c1(C2C(NC(c3cn(C4C(OCC)COC4)nn3)=O)CCO2)ccc(Cl)c(F)c1 c1(C(C)C)ccc(C#N)c(NC2CN(C(=O)C(C)C3CCC3)C2)n1 C1(OC)(NC(C2CC(C)(C)CO2)=O)CCN(C(=O)CNC(=O)CNC(C)=O)C1 C(C(F)(F)C(C)(C)O)NC(C(CCC)NC(c1ccnn1C)=O)=O c1(N2C(C)(CNC(c3ccc(CC)s3)=O)CCC2)ncnc2cc(C)[nH]c12 C1(C(=O)NCCCN(C(=O)Cc2ccc(F)c(Cl)c2)C)CCCS(=O)(=O)N1 c1(C2C(NC(c3cccc(C4C=CC(C(=O)O)C4)c3)=O)C2)c(F)cccc1Cl Cc1cccc(C(=O)NCCCC(C)NC(=O)CCOCC2CCCO2)c1N C1(CN(C2CC(CC(=O)N(C3CCCC3)CC)C2)C)CCN(C(C)=O)CC1 N1(C(C(COC)C)=O)CCC(C2(NC(c3ccc(N(C)C)cc3)=O)CC2)C1 c1(NC(C=CC)=O)cccc(Br)c1OC(C)COC(=O)C(C)C CN=c1cc(C(N2CCN(C)CC2C(=O)NCC2(C)CNC(=O)O2)=O)cc[nH]1 Cc1c(Cl)ccc(C(=O)N(C)CC2CCCCN2C(C2CCOC2C)=O)c1O C1(CCC)CCCCN1C(=O)C=CCNC(=O)C(O)COC c1(C(N2CC(O)(CNC(C(c3ccccc3)N(C)C)=O)C2)=O)cc(O)cc(Cl)c1 Cc1cc(C)c(-c2ncc(C(N3CCN(C)C(=O)C3)C(=O)NC(C)C)s2)c(C)c1 C(=O)(CCC(=O)N1CC(NC(C2CC(N3CC(O)C3)C2)=O)C(CC2CC2)C1)NC C1(OC)(CNC(c2cc(F)n[nH]2)=O)CN(C(c2cc[nH]c2C2CCC2)=O)C1 C1(NC(c2cncc3sccc23)=O)CC2CCC1N(C(=O)C1=CCSC1)C2 CCCC(C(=O)NCC1CCCSC1)NC(=O)CCC1CC(COC)C1 Cc1ccnc(C(N2CCC(N3CCN(C(c4cc(C)[nH]c4C)=O)CC3)C2)=O)n1 CC1=NNC(=O)C1CC(N1CC(C(C)NC(=O)CCNC(=O)NCC2CC2)C1)=O N1(C(c2ccc(C)s2)=O)CCCC(C2CN(Cc3ccc(O)cc3O)C2)C1 C1(C(=O)NC(CC#C)CCOC)CC(C)(C)CCN1C(c1ccc(C)cn1)=O C1(NC(=O)CC2CCOCC2)COC2(CCN(S(=O)(=O)c3ccc(F)cc3)C2)C1 N1(C(C2(COC)CC2)=O)CC2CCCC(NC(c3ccc(C)nc3OC)=O)C2C1 N1(C(c2nc(C(C)NC(C(C=C)(F)F)=O)oc2)=O)CCCC(OC)CC1 CCS(=O)(=O)C1CCN(C(c2cccnn2)C(=O)NCc2cccc(Br)c2)C1 c1(C(=O)NCC(C)(C2CC2)NC(=O)COC2CC=CC2)ccc(Br)c(N)c1 C(CCCC(=O)NC1C(C)CCC1C)NC(Cc1ccn(CC)n1)=O C1(CNC(C(C)O)=O)CN(C(c2cccc(NS(N)(=O)=O)n2)=O)CC12CC2 C12(C(N(CCCC)CCCC)=O)CC1CCN2C(c1scnc1CC)=O C(=O)(C(CC(F)F)NC(=O)Cn1nccn1)NCC(C)(C)CCO c1(C(=O)NC2CN(C(c3c(CCC)n(C)nc3)=O)C2)cnc(C)c(C#N)c1 c1(NC(c2c(OC)ccc(Br)c2)C2CC2)cccc(C#N)c1O C1(NC(CC(n2c(CC)ncc2)C)=O)CCCC2CN(C(C3(C)CC3)=O)CC12 n1(CC(=O)NCC2(NC(CC)C(=O)N(C)CCSC)CC2)cc([N+](=O)[O-])cn1 CCCCCCC(=O)N1CCCC1C1C(C(=O)N(CCCO)CC)C1 Cc1cc(C(N2CC(NC(=O)CC3(NC4CC4)CCC3)C(C)C2)=O)nn1C(C)C CC1=C(C(=O)N2CCN(C(c3cn(CC(N)=O)nn3)=O)CC2CF)CCS1(=O)=O c1(C(N2CCC(CC(=O)NCc3nc(CC)sc3)C2)=O)ccc2ncnn2c1 N1(C(C2N(C(Cc3ccc(OC)cc3)=O)CC(C)C2)=O)CCC(O)(C(=O)OC)CC1 c1(OC(C)C(N2C(C3(N(C(=O)C=CI)C4CC4)CC3)CCC2)=O)cccnc1 C(=O)(CS(=O)(=O)Cc1cccc(Br)n1)NC1(CC(=O)OC)CC1 N1(C(c2cc(CC)ccc2F)C(=O)NCCOCC)CC2CCC(C1)C2C#N N1(C(C2CCCC(N(C)C)C2)=O)CCCCC(NC(C23CC(F)(C2)C3)=O)C1 c1(C(N(c2c(C)cccc2)C(=O)C(C)NC(C)C(C)C)=O)ccc([N+](=O)[O-])cn1 C1(C(=O)OC)(CF)CCN(C(C2CC(C)CN2C(=O)CC2CC3C=CC2C3)=O)C1 C1(C(N2CCC(CN(C)C(c3cncc(N)c3)=O)C2)=O)C2CCC1(C)C2(C)C C(=O)(C1=CCCCCC1)N1C(C)(C(C(=O)Nc2c(C)ncc(Cl)c2)CN(C)C)CC1 N1(C(CSC(C)(C)C)=O)CCOCC(NC(=O)C(c2cncn2C)O)C1 N1(C(C2(C#C)CCCC2)=O)CCC(C2CCN(C(C3CC(O)C3)=O)C2)CC1 C1(CN(C(C(C)CO)=O)C2CC2)CCCN(C(=O)COc2cccc(Br)c2)C1 N1(C(CCn2ccc(C)n2)=O)CCC2(CCN(C(=O)C(C)c3ccn[nH]3)C2)C1 C1(C)(CNC(c2c(C)nc[nH]2)=O)CCCN(C(=O)C(c2cc(Cl)cc(Cl)c2)=O)C1 C1(C)(C(=O)NC(c2n(CC)ncn2)C)CN(C(=O)C(C)S(C)(=O)=O)C(C)(C)C1 C1(C(=O)NCC(C2CCN(C(=O)CC3CC(=O)C3)CC2)(C)O)CC(=O)NC(=O)N1 C(C(C)(C)CC(=O)NCC1CCN(CC2(C#N)CC3CC3C2)CC1)OC CCC(C)(C(=O)NC1CCCC1NC(=O)COc1cccc(C)c1)OC c1(CN=C(NCCSC)NCC2(O)CC3CCC(C3)C2)c(C)oc2ccccc12 c1(N(C(C(C)=CC)=O)C2CC2(F)F)ncc(-c2ccccc2F)cn1 c1(N(C)C)ncc(C(=O)NCC2CCN(C(=O)Nc3cccnc3)C2)cn1 c1(CN(C)CC2CN(C(C3CC3F)=O)C2)cc(Cl)cnc1F N1(C(C2CCC(C)(C)C2)=O)CCCC2CN(C(c3cc4c(s3)CCC4)=O)CCC12 c1(C(=O)NCCCCC(C)NC(c2cncc(C)c2)=O)c(N)c(F)cc(F)c1F C1(C(=O)NCCC(C)N(C(c2c(C)c[nH]c2)=O)C)CCC(O)CC1 C1(C)(C(=O)NCC(C)NC(CC=C(C)C)=O)CCCCC1(F)F C(c1cnn(C)c1C)=CC(C)NCC1CCCN1C(=O)C(C)n1ccnn1 C1(C(=O)NCC2C(CNC(c3cc(C(CC)C)no3)=O)C2)CCCCC(=O)N1 c1(OCc2ccc(OCC)cc2)ccc(Cl)c(O)c1S(=O)(=O)NNC=O c1(C(=O)NC2CC(CNC(CC3CC(OC)C3)=O)C2)csc(-c2cn[nH]c2)n1 C1(CC(=O)Nc2[nH]nc(CC)n2)CCC(=O)N(CCNC(=O)NC(C)C)C1=O C(=O)(C(C(C)(C)C)N(C)C)NC1(CO)CCN(C(CC=C)=O)C1 C1(CNC(CCc2c(C)n[nH]c2C)=O)CCN(C(=O)CC(C)F)C12CC2 c1(N(CCC)CCNC(c2csc(C(C)C)n2)=O)ncnc(C)c1F C1(CC)CC(C(=O)NC(C2CN(C(c3csc(C4CC4)n3)=O)CCO2)C)CCO1 C(=O)(C#Cc1cccc(Cl)c1)OC(c1c(F)cccc1F)C c1(CC)nn(C)c(CNC2C3CCC(O3)C2C(N)=O)c1Cl CC#CCCCCNC(C12CC1CN(C(=O)CCC(C)N(C)C)C2)=O C1(c2c(C)cccc2)CN(C(=O)C(=O)NCC2CCCS(=O)(=O)C2)CC(=O)N1 C1(C)(NC(CN(C(C(n2ccc(C)n2)C)=O)CC(C)C)=O)CCC2(CC1)CC2 C(C(C)(CC(=O)NCC1(c2ccccc2)CCCC1)C(F)(F)F)N(NC)C c1(C(N2C(C(=O)NCc3cc(CC)[nH]n3)CC2)=O)ccc(O)nc1 CC(C)C#CC(=O)N1CCC(CN(CC(c2ccc(Cl)cc2)O)C)C1 c1(C(NOCc2cn(Cc3ccc(OC)cc3)nn2)=O)cc(C#N)c[nH]1 C=CC(C)C(C)C(=O)NCC1CC(NC(c2csc(CN3CCCC3)n2)=O)C1 C1(C(N2C(CCC(=O)NCCCC3CCCCC3)CCC2)=O)CCC(F)(F)C1 Cc1c(O)ccc(C(=O)NC2CCC2NC(c2cc(O)nn2C)=O)c1C CC(CC(=O)NC1CC(C(F)F)C1)C(C)(C)NC(=O)CCCC1CCC1 CC(CC(Cl)Cl)C(=O)NNC=O.C(CF)O CCCCCCC(=O)NC1CC(CNC(=O)Cc2csc(C(C)C)n2)C12CCC2 c1(C(N2CC3C(C(=O)NC4(C(F)(F)F)CC(=C)C4)(C3)C2)=O)cccc(C#N)c1 C12CCCC(C1)NC(=O)C13CC(C1)(C3)C(=O)N(CC)C2.c1(OC)ccc(C)cc1 C(C(C)C)(C(O)C(=O)N(C1CC2CCC(C1)N2C(=O)C(C#N)C(C)C)C)OC C1(C(=O)NC(C(=O)O)CO)CCc2c(nnn2CCO)C1 C1(NC(CC)=O)CC2CCC(C1)N2C(C1C=CCN(C(C)=O)C1)=O.C(C)(C)(C)O Cc1c(F)ccc(C(N2CCN(C(c3cc[nH]n3)=O)C3CC23)=O)c1C#N CC1CCN(C(c2cccc(C3CC3)c2)=O)CC1CC(=O)NOC(C)(C)C C(=O)(C(CC)C(F)(F)F)NCC(CC=C)NC(c1ccc(C#N)cc1F)=O N1(C(C2=NOC(C)(C)C2)=O)C2CCCC1CC(NC(C13COCC1C3)=O)C2 N1(C(CCSCC)=O)CCCC(C2CN(C(c3ccc(F)c(Cl)c3N)=O)C2)C1 c1(CC)c(C(N2CCC(N(C(=O)CC3COC4CC3C4)CC)C2)=O)cccc1F Cc1c(-n2cc(C(C)N(C(=O)CN(CCS(C)(=O)=O)C)C)nn2)cccc1O CN1CCN(C(c2ccc(C(N3CC(n4ccnn4)C3)=O)o2)=O)C(C2CC2)C1 c1(C(C(=O)NC(c2cnn(C)c2)C(=O)NCCCOCC)=O)ccc(O)cc1 C1(C(=O)NCC2(CC(=O)OC)CC2)CC(O)CN1C(C1CN(C(C)C)C1)=O CCC(C)(C)CC(=O)NC1CC(F)(CNC(c2onc(OC)c2Br)=O)C1 C12(NC(CCCC=C)=O)CCC(C(N3C(C)CCCC3C)=O)(CC1)C2 C1(N2CCC(NC(=NCC(C)OC)NC3CC3)CC2)(N(C)C)CC(C)CC(C)(C)C1 Cn1nnc2cc(C(=O)NC3CCCC(CNC(c4ccco4)=O)C3)ccc12 c1(C(=O)NCC2(NC(c3ccc(Br)cc3O)=O)COC2)[nH]nc2ncccc12 C1(C(=O)NC2CCN(C(C)C)C2)CN(C(C2(CC3CCC3)CC2)=O)CC(C)(C)C1 C1(C(C2CCC2)N(CC(=O)NCC(COC)O)C)CCOCC1 C(C)(C)(CC(F)C(=O)Nn1cnnc1)NC(C1CCC2C(C)(C)C1C2)=O c1(C(c2nnnn2C2CCOC2)NCCn2c(C)ncc2)cc(Br)cnc1F N1(C(CC(=O)OC)=O)CCC2(CC1)CCN(C(c1ccnc(OC(C)C)c1)=O)C2 N1(C(COCCC(C)C)=O)CC(CCNC(C2(O)CCC2)=O)OC(C)C1 c1(C(N(C2CN(C(=O)CC(O)c3ccccc3)C2)C)=O)ccc(N)c(F)c1F Cc1cc(F)c(C(N2CCCC(F)(CNC(C3C4CCOCC34)=O)C2)=O)c(Cl)c1 c1(C(N(CCN(C(=O)CCc2cccnc2)CC)CC)=O)nocc1Br c1(CC)ccc2c(c1)C(CCN1CCCCC(CO)C1)C(=O)N2 c1(COC(c2n(C)ncc2)=O)ccc2c(=O)[nH]ccc2c1 C(=O)(C(F)C(C)(C)O)N1CCCC(N2CCN(C(C(C(C)C)SC)=O)CC2)C1 c1(C(C(=O)OCC)N(C)CC)sccc1OC.c12cnc([nH]1)CC(=O)N2 c1(CCNC(=O)CNC(=O)CCc2ccc(Br)cc2)cnc2ccccc2c1 CN1CCN(c2ccc(CN3CCC(F)(C(N4CCC(F)C4)=O)C3)s2)CC1 c1(CC)noc(C)c1C(=O)NC1CCC(N(C(=O)C=Cc2cnn(CC)c2)C)C1 c1(C2C(C(=O)NC(CN(C(=O)COCC3CC3)C)(C)C)CC2)ccccc1Cl C(CNC(C1(c2cscn2)CC1)=O)(CC(C)C)NC(c1nc(CC)oc1)=O c1(-c2cn(C3C=CCC(C(N4C(C)CC(F)(F)C4)=O)C3)nn2)cc(F)c(N)cc1F c1(C(=O)NC2C(NC(C(C)(C)CC#N)=O)CCCC2)c(Cl)ccc(Cl)c1Cl C=Cn1ncc(C(N2CCCC2C(=O)NCCn2cnnc2)=O)c1N C1(NC(C(C)Sc2ccc(C)cc2)=O)CCCN(C(=O)CC2CCC(C)C2)CC1 C1(C(N(C)Cc2ccccc2O)=O)CC2(CC2)CN1C(C1CCS1(=O)=O)=O c1(C(=O)NCCN(C(C2(C)CCCN2)=O)C2CC2)ccc(Cl)cn1 C(c1ccc(C)cc1)=CC(=O)NCC1(NC(C2C(CC)CCC2)=O)CCOC1 C12(C(=O)NC3CCN(C(C=C(C)c4cccnc4)=O)C3)CC1COC21CCC1 N1(C(c2ccc(C)o2)=O)CC2CC(NC(=O)Cc3cnn(C(C)(C)C)c3)CC2C1 C12(CNC(C(=O)NC3CC3)=O)CCCC1CCN2C(C1CCC=CCC1)=O c1(NC(C#C)C2CCC2)ncn(C)c1C c1(OC)c(C(=O)NCCCC(C)NC(c2c(N)cccc2Cl)=O)ccnc1F c1(OC(C)C)cccc(C(=O)NCC2(O)CN(C(C3CC(C(F)(F)F)C3)=O)C2)c1 C(=O)(CCC(C)NC(=O)C(C)N1CCCC1)NCC1(CC(C)C)CC1 Cc1ncc(CO)c(CN2CCC(C3(C(=O)NC)CNC3)CC2)c1O c1(C(N(C(CCNC(C2C(C)CC=CC2)=O)C)C)=O)cc2scc(Cl)c2[nH]1 Cc1nn(C)c2nc(C(N3CC(NC(=O)C(F)C(C)C)CC(C)C3)=O)ccc12 c1(C(c2nnnn2CC(F)F)NCCC(=O)NC)ccc(N(C)C2CC2)cc1 c1(CC)nc2sc(C)cn2c1C(N1CCC(NC(=O)C(C(C)C)N(C)C)CC1)=O C12(NC(C(CCCC)=O)=O)CCCC1CN(C(c1c(CO)n[nH]c1C)=O)C2 C1(CNC(c2cn(CC)nc2)=O)CN(C(C2(O)CCC2)=O)CCC1C C1(CNC(N2C(C)CN(CC)C(C)C2)=O)CC2(CCOCC2)CO1 N1(C(C(C)=C(CC)C)=O)CC=CC1(C(=O)NCCn1ccccc1=O)COC CC1CCN(C(=O)Cn2cccn2)C(C(=O)NC2CC(C)(C)C2)C1 c1(C(=O)NC(CCCC)CNC(=O)CNC(C2CCC2)=O)cc2c(s1)CCCC2 C(C(C)(C)C(=O)NCC12CC1CN(C(C1CC1c1ccccc1F)=O)C2)OC CC1(C(=O)NCC(C2CCCC2)NC(=O)C(O)C2CC2)CSC1 N1(C(C(CC)C(F)(F)F)=O)CCCC2(C1)CN(C(C1(C)CC1)=O)CCO2 C(=O)(CCC(=O)NC(C1CCCC1)CNC(=O)Cc1n[nH]c(C)n1)NCC N1(C(c2nccs2)=O)CCC(C2CN(S(=O)(=O)CCCCl)C2)CC1 C1(NC(Cc2ccc(CC)cc2)=O)CN(C(=O)C(C)(Cl)Cl)CCC1C(F)(F)F C1(CC(=O)N(CC(C)OC)C)CN(C(C2(OCC)CCCCCC2)=O)CC1(C)C CC1C(NC(c2n[nH]c(C3CC3)n2)=O)CCCN1C(=O)C=CC1CCCC1 N1(C(Cc2cc(C)nn2C)=O)CCOCC(F)(CNC(c2conc2C)=O)C1 Cc1nn(C)c2c(N3CC(C)S(=O)C(C)C3)nc(=NCC3OCCO3)[nH]c12 c1(SC)cc(C(=O)NCCC2CCC(NC(=O)CCC3CC3(F)F)C2)c(C)o1 c1(C(N2CC(NC(=O)Cc3ccccc3)C(O)C2)=O)ccc([N+](=O)[O-])nc1 c1(C(N2CC(NC(Cc3c(C)n[nH]c3)=O)C2)=O)cc(-c2cccc(Cl)c2)n(C)n1 c1(NCC2(CC)CCCC2)[nH]c(=NCCCOCC2CC2)nc2ncn(C)c12 C(=O)(CS(=O)(=O)CCC)NC(CC)CNC(C1(c2ccccc2)CCCCO1)=O c1(NC(C2(O)CCC(C)CC2)=O)cc(Br)cc(I)c1F c1(C(=O)OCC)c[nH]c(C(=O)NC2CC2c2cn(C(C)(C)C(=O)O)nn2)c1C C(=O)(CCCC(=O)NCC1(O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1)OC C(C(F)(F)C(=O)NC(c1cn(C)nn1)C(=O)N(C1CCC(C)CC1)C)N(C)C N1(C2(C(=O)COC(C)C)CC2)CCCC(C(=O)N(CCCN(C)C)CCO)CC1 Cc1nn2ccccc2c1C(=O)NCCCCN(C(=O)CCC(C)C=O)C C1(C(C)C)OCCCC1C(=O)NCCC1CSCCN1C(c1ccc(=N)[nH]c1)=O c1(COC)ccc(C2(CCCN3CCC(OC)CC3)CCO2)cc1 N1(C(c2cncc(OC)c2)C(=O)NC2(C)CC2)CCCOC(C)C1 CC1(C)CC(NC(c2ccccc2OCC(N)=O)=O)CN1C(C1CCC(=O)N1)=O C(=O)(C1=CC(C)(CC)C1)N1C(CC=C)(C(=O)NCC2CC23CCC3)CCC1 Cc1sc(O)nc1C(=O)NC1CN(C(=O)C(F)=CCCF)CC1C(F)F C1(C(=O)NC(C(C)NC(c2cnnc(O)c2)=O)CO)CC2CCC(C1)C2O C=C(Cl)C(C)(C)C(=O)N1CC(N2CCN(C(=O)CSc3nncn3C)CC2)C1 N1(C(COCCCC)=O)CCC2(CC1)C(NC(=O)C(C)C(F)F)CS2(=O)=O c1(C(=O)NC(CCCC)CNC(=O)C(C)(C)N(C)C)cnc(O)n(C)c1=O Cc1c(NCc2c(Cl)cccc2Br)nc[nH]c1=NCc1ccnn1CC(F)F C(=O)(CC(CCCC)NC(c1cc(O)cc(F)c1)=O)NCC1(CCC=C)CC1 c1(N2CC3CC(C)C(=O)N3CC2)nc2ccsc2c(=NC(C)COCC(F)(F)F)[nH]1 c1(C(=O)NCC2(C(=O)OCC)CCC2)ccccc1-n1ccnn1 C(=O)(C1c2c[nH]nc2CN1C(C1OC2CCC1C2)=O)N(C)Cc1onc(C)n1 C1(F)(CNC(C(C)OCCC#C)=O)CCCN(C(=O)C(CC)C(C)C)CC1 CC1(O)CCN(C(=O)CCC2CCC(NC(=O)CN3CCCCC3)C2)CC1 C1(C(=O)N)CCC2CC12COC.C(=O)(CC(=O)N)N1CCCC1.C(C(F)F)OCC N1(C(c2cnc(CC)s2)=O)CCC(C)C(NC(=O)C(=O)Nc2cccc(C)c2)C1 N1(C(Cn2c(C)ccn2)=O)CCCC(C2CCCN2C(c2cc[nH]n2)=O)C1 CCCCC(C)C(=O)N1CCCC(C)(NC(c2cnc(O)cc2O)=O)C1 C1(NC(=O)C(O)C2CCCC2)CC2CC(NC(=O)CCC3CC(F)(F)C3)C1C2 N1(C(C(=O)NCC2C(CNC(C3CC(OC)C3)=O)C2)CC)CCc2ccccc21 C(=O)(CCS(C)=O)N1CC(N(C(C2C(c3scc(C)n3)C2)=O)C)C1 C=CC1CN(C(c2csc(S)n2)=O)CC1NC(c1cc(CO)n(C)n1)=O CC(C)CS(=O)(=O)CCC(=O)NCC(O)CN(C(=O)CC1(O)COC(C)(C)C1)C c1(C(N2CCC(CCNC(C3(n4nccn4)CC3)=O)C2)=O)cc2ccccc2o1 C(=O)(C(F)(CNC(C1CC(CF)C1)=O)C(C)C)NCC1(C)ON=C(C)C1 Cn1c(C(=O)NCC2CCCC(NC(C3CN(C4CCC4)C3)=O)C2)cccc1=O CCC(CC(=O)N(C(C)C)C1CC1)NC(C1CCC(C)CC1)=O N1(C(C2N(C)C(=O)CC2)=O)CC2CN(C(c3ncc(Br)cc3O)=O)CC2C1 CC(CCCNC(C1CC1(C)C)=O)NC(=O)C(F)Cc1ccccc1 c1(C(N2CCN(C(Cc3cc(C)on3)=O)C(C)CC2)=O)c(C)nn2c1NCCC2 c1(C(=O)NC2CC3CN(C(c4cncnc4)=O)CC3C2)cc2cccc(Cl)c2[nH]1 CC(C)C(F)(CNC(c1cc(O)cs1)=O)C(=O)N1CC2CCCCC12C C12(C(=O)NC(C)C(F)(F)F)C(NC(=O)CN3CCNC(=O)C3)C3CC1C2C3 c1(CNC(C(C)OCC=C)=O)cc(C(=O)NOCCCF)co1 CC1(C(=O)NCC=CCNC(=O)CC(c2cc(Cl)cc(Cl)c2)O)CCNC(=O)C1 c1(C(N2CCC(N(C(C(C)SCC)=O)CC)C2)=O)c(O)nnc(CC)c1CC c1(CC)[nH]nc(Cl)c1C(=O)NC1CC(NC(c2cc(C(C)(C)C)nn2C)=O)C1 c1(C(=O)NCC(CNC(C2CC(C)(O)C2)=O)F)ccc(-c2coc(O)n2)cc1 c1(C(=O)OC)cc2n(n1)CC(OC(c1ccnn1C1CC1)=O)CO2 C(CC(C)C(=O)NC(CSCC)C(=O)NCCCCN=[N+]=[N-])=CCC N(C(=NCCc1ccc(Cl)s1)N1CCC(F)(C#N)C1)C1C(C)CCC1 C(=O)(C1=CCCOC1)NCC(CN(C(c1ccn(CCOC)n1)=O)C)(C)C C1(C(=O)Nc2nccs2)CC12CCN(C1CC1)CC2.c12ccc(C(F)(F)F)c-1c2 N1(C(CC(C)SC)=O)CCC(C)(C)C1CNC(c1ccc(-c2ccc(C)o2)s1)=O Cc1cc(Cc2ccccc2)oc1C(=O)NCC1CCN(C(C23CC(O)C2C3)=O)C1 C12(C(N(OC)C)=O)CCC(F)C1CC2.N12CCCC1CC1(CC1)CC2=O.C1(C)CC1 c1(C(=O)NCC2C(NC(C3(C)CS(=O)(=O)C3)=O)C2)cc2cccc(Cl)c2o1 N12CCN(CC1)NCC2CC.c1(NC(C2CC(C(N)=O)C2)=O)ccc(OC)cc1 N1(C(C#CC(=O)N(C)C)=O)CCC(NC(C2CC(=O)N(C)C2)=O)CC(O)C1 CCC1=NOC(CC(=O)NC2CN(C(=O)CCCCN(C)C)CC2SC)C1 n1(C(C(=O)OC)C)nnnc1C(c1nc(C)cs1)NC(=O)CCCc1ccccc1 N1(C(CNC(=O)CN2CCN(CC(F)(F)C(F)(F)F)CC2)=O)CCOC2CCCC12 Cc1sc(C(=O)NC2CC23CC(NC(c2ccc[n+]([O-])c2)=O)C3)cc1[N+](=O)[O-] C1(CC#C)(C(=O)NCC(C)C(=O)NC2CN(C3CCC3)C2)CCCO1 C(=O)(C1=C(C2CCCOC2)N(C)C(=O)NC1c1cc(OC)ccn1)OCC CCS(=O)(=O)CC(=O)N(CC(O)CN(C(=O)C(c1cccc(C)c1)(F)F)C)C c1(C(=O)NCC(C)N(C(CCOCCOC)=O)C)coc2c(Cl)cccc12 Cc1cc(=NC(=O)CC2SCCN2C(C(C)(C)C)=O)[nH]n1C(C)C1CC1 C1(C)(C(=O)NC)CCCN1C(=O)COC1CC(NC(C2CCOC2)=O)C1 C1(C(=O)NCc2c(C)nccc2)CN(C(=O)CC2CCCCCC2)CC1C#N C1(C(C)NC(C(C)OCCC(C)C)=O)CCCN1C(=O)CO CC1CCCc2nc(C(=O)NCC3(NC(C4CCCC4C)=O)CCCC3)cn21 c1(C(=O)NCC(CO)NC(Cc2ccc(C(C)=O)s2)=O)cccc(CCC#N)c1 Cc1nc(NCCN2CCC(P(C)(C)=O)C2)cc(=NC(C)c2ccco2)[nH]1 c1(CC)cc(NC(C2CCCCC2CNC(C2CCC(=O)C2)=O)=O)cc(F)c1 Cc1cccc(N)c1C(=O)NCC(O)CNC(C1(C)CCC12CCC2)=O c1(OCC)ccc(C(=O)NC2C3CC2N(C(=O)CCN(C)C)C3)cc1C C1(CNC(C(c2n(C)ncc2)O)=O)CC(C)(C)CN1C(=O)CCOCC(F)(F)F c1(CC)nc(C)ncc1C(N1CCN(C(=O)CC2(COC)CC2)C2CC12)=O C1(O)(CNC(C2N(C(C(C(C)C)C3CCC3)=O)CC(O)C2)=O)CCN(C)CC1 c1(CNC(C2CN(C(=O)C(C)C(C)(C)C)CCO2)C)cnc2n1CCCCC2 N#Cc1ccc(Br)c(C(N2CC(c3cn(-c4nc5ccccc5[nH]4)nn3)C2)=O)c1 C1(NC(C(C)n2ccnc2)=O)CCN(Cc2cncc(Br)c2)CC1(C)C C(=O)(C(CCC(C)C)NC(C)=O)NCCc1c(CNC(C(CCC)C)=O)nco1 C(N=c1[nH]c(=NCC2(C)CC2(C)C)c2c(ncn2C)[nH]1)c1c(CC)noc1C c1(C(=O)OC)coc2c1CN(C(=O)Cc1nn(C)cc1[N+](=O)[O-])C2 c1(C(=O)COCC2(C(N3CC(C=C)(O)C3)=O)CCC2)cc(C)cc(C)c1 C(=O)(C(C)S(=O)(=O)C(C)C)N1C(CNC(c2cccc(CC)n2)=O)CN(C)CC1 Cc1ccc(C(=O)NCC(N2CCC2CNC(=O)C(F)=C2CCC2)=O)cc1 C#CC(C)(C)C(=O)NC(CC)CC(=O)NCC1CC(N2CCCC2)C1 C1(N(C(=O)CNC(=O)CC)CC)CCCN(C(=O)CCCN2C(=O)CNC2=O)C1 CCC(CC)C(C)C(=O)NC1CN(C(c2c(C(F)(F)F)cnn2C)=O)C1 Cc1cc(C(C)C(=O)OC(c2ccc(F)c(F)c2)C)cc(C)c1 C(=O)(C#CC1CCCCO1)N(CC(O)CN(C)C(c1ncc[nH]c1=O)=O)C N1(C(C(C)OCCCC)=O)CC2C(CN(C(=O)CCc3cn(C)cn3)C)C2C1 N1(C(Cc2cn(CC)nc2)=O)CCCC(C)(C(=O)NCC2CN(C)CCO2)C1 CCCCC(CCC)N=c1[nH]c(=NC(C)c2cc(CC)no2)c2c(F)cccc2[nH]1 C(=O)(C(C)C(O)C(C)C)N1C(CCNC(c2c(C)cc(CC)o2)=O)CCC1 Cc1ccc(C(N2CCCC(C)(NC(c3coc(C(F)F)c3)=O)C2)=O)nc1C C1(CNC(=O)C(C)OC)(CO)CC2CC2C1.C1(CC#C)(C(=O)NC)CC1 C=CCCCC(C(=O)N(C)CC1CCOCC1)NC(=O)C(C1CC1)OCC CCCCCC(=O)NCc1cccc(CN(C(=O)Cc2nn(C)cc2Cl)C)c1 C1(C(=O)NCCCCNC(=O)CCC(=O)c2ccc[nH]2)CCC(N=[N+]=[N-])C1 C1(CNC(C2CCCC2C(N2CCCC(C(F)F)C2)=O)=O)CC(C2CC2)=NO1 C1(C(N2CCCC(N(C(CCSCCC)=O)C)CC2)=O)CCCC(F)(F)CC1 C1(c2n(C)ccn2)CN(C(=O)CC2CC2C2CC2)CCN1C(=O)COCC1CC1 C1(C)(CC)C=C(C(=O)NCC2CC(O)CN2C(c2cc(C(C)(C)C)n[nH]2)=O)C1 CC1CCC(NC(C2(CO)CCOCC2)=O)CN1Cc1cnn(C)c1 N1(C(C(C)OCCN(C)C)=O)CC2CC2C1CNC(=O)Cc1ccon1 C1(NC(C2CCC(=C)CC2)=O)CN(C(c2ccc(N)c(C)c2)=O)CC(C)(C)C1 C(=O)(C1Cc2ccccc21)N(CC(CO)(CO)NC(C(C)OCCN(C)C)=O)C c1(C(=O)NCC2(COC)CN(C(c3[nH]cnc3C#N)=O)C2)oc(C)cc1C c1(C(N(CC(CN(C(C(c2cccc(Cl)c2)C)=O)C)O)C)=O)cccnc1O C(=O)(C(C)CC(=O)c1ccccc1)NC1(CC=C)CC2C=CC1C2 c1(C(=O)NC(CC)(C)CNC(c2ccoc2C)=O)c(O)cnc2ccccc12 N1(C(C2(CC)CCCC2)=O)CCC(NC(c2ccn(C(C)C)c2C)=O)C(O)C1 c1(C(C(=O)NCCCF)N(CCC#N)CCC)cccc(CO)n1.C1(CN)CC1 c1(CCNC(C2C(CCOC)C2)=O)ocnc1CNC(C1CC1Cl)=O C(c1cc[nH]c1)=CC(=O)NC(C(=O)NCCC#CC)C1CCOC1 c1(N2CCCC(CCS(N)(=O)=O)C2)nc2cc(Br)ccc2s1 N1(C(C(COC)OC)=O)CC2CCCC(NC(=O)CN3CC=CC3)C2C1 C(=O)(CC(C)C(F)(F)F)NCC1C(NC(C2N(C(C)=O)CCC2)=O)CCCC1 N1(C(c2n(COC)ncc2)=O)C2CCC1C(C)C(NC(c1n[nH]cc1C)=O)C2 c1(CCC(=O)OC)c(F)cccc1F.C1C(CCC)=C(F)C(=O)N1CCCN C1(NC(C=Cc2n(CC)ncc2)=O)CCN(C(C23CCCC2C3)=O)C(C)C1 N1(C(c2c(OC)c[nH]n2)=O)CCN(C(C2CC(c3ccccc3)CO2)=O)CC1 C1(NC(Cc2nc(C)sc2C)=O)CN(C(C2(C)CCCCC2)=O)CCC1C c1(OC)ccc(Cl)c(NC(C2CCN(C(=O)C(c3ccccc3)=O)CC2O)=O)n1 Cc1c(C(=O)NCC2CCC(NC(c3ccno3)=O)CC2)[nH]c2cc(Cl)ccc12 C1(N(C(=O)CC2CC=CC2)C)CCCN(C(c2ccc(C(O)CF)cc2)=O)C1 N1(C(C=Cc2ncn(C)c2)=O)CCC2(CC1)CC2C(=O)O N1(C(C(CC)SC)=O)CCCCC1CCN(C(=O)CCCOC(C)(C)C)C c1(C(c2ncn3c2C(C(=O)O)C3)=O)cc(C(F)(F)F)c(Br)cc1[N+](=O)[O-] N1(C(CCCC#C)=O)CCC(CO)C(NC(c2cc(C)nc(C(C)(C)C)n2)=O)C1 C1(C(=O)NC(C(=O)OC)CCF)C2CC3C(C2NC(C2CCCCC2(C)C)=O)C13 c1(C(=O)Nc2ccc(C(C(C)(C)C)(C)C)cc2)nc(C(F)(F)F)n2ccccc12 N1(C(COC)=O)CCC(O)(C(C)CNC(C2(C(N)=O)CCC2)=O)C1 C(=O)(C(C)(C)CC(C)C)N1CCC(n2cc(C(c3ccccc3)COC)nn2)C1 N1(CCCNC(=O)C=CCOC2CCCCC2)CCN(C(C2CCCS2)=O)CC1 c1(C(=O)NC2C(C=C)CN(C(c3cnc(C(C)O)s3)=O)C2)cnc(O)n(C)c1=O c1(C2(NC(C3C(C=C(C)C)C3(C)C)=O)CCCC2)cccc(Br)c1Cl C1(C(N2CC(N(CC=C)C)C2)=O)CC2CCC1N2C(=O)CC(C)CN(C)C c1(C(N(CCCNC(=O)C(C)SC)CCC)=O)cccc(CC)c1 C1(C(=O)NC(CC=C)C)CCCN1NC(=O)C(C)N1CC(=O)NC1=O C1(NC(c2cnn(C(F)F)c2C2CCCC2)=O)CC2(C1)CC2NC(C1CCC1)=O C1(C(=O)NC2CC3CC(NC(C4CCC=CO4)=O)C3C2)CC2(CCOCC2)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCC(C)N(C(=O)CC2CCC(F)(F)CC2)CC1 C(=O)(CC(=O)NC1CC(NC(=O)C(=O)NCCC2CC2)C1)NCC#C c1(CC(CNC(=NC)NCC(F)F)CO)c(F)cccc1F CC1CC(NC(=O)CCC2CCC2)CN(C(=O)CC2CC2)C1 N1(C(C(CCOC)C)=O)CC2C(NC(c3cnn(C(F)F)c3)=O)CS(=O)(=O)C2C1 C(C(C(=O)OC(c1ccc(Br)cc1)C#N)C(F)(F)F)OC S(=O)(=O)(c1cccc(OC(F)F)c1)NS(=O)(=O)CCBr.C12CCN(C1)C2 C(=O)(CCN=C(NCC(F)F)NCCn1cncn1)N(C)Cc1ncn(C)n1 N1(C(C(CC)OCC)=O)CCC2(CCCN(C(c3ncc4n3CCCC4)=O)C2)C1 C=CCCCC(C(=O)N(Cc1ccccc1)OC)NC(=O)Cc1coc(C)n1 n1(C(=O)OCC)nccc1[N+](=O)[O-].C12CN(C1)C(=O)N2 c1(C(N2C(C(N3CC(C)C3)=O)C3CC(F)C2C3)=O)ccc2ccc(Cl)cc2n1 C1(CC2(Cn3cc(CNC(C4N(C)CCCC4)=O)nn3)CC2)CCOC(C)(C)C1 c1(NC2(CNC(C(C)(C)OC)=O)CCCCC2C)ccc(F)cc1[N+](=O)[O-] Cc1cccc(Cl)c1C(=O)NC1(CNC(=O)CC2CC3CCC2CC3)CCC1 ClC=CCN=c1nc2sccc2c(NCC2CSCCSC2)[nH]1 C(=O)(NNc1ccc(C#N)cc1C(F)(F)F)NC(C1CCC(F)(F)CC1)CC c1(C(=O)NCCN(C(C(CC=C)CC)=O)C(C)C)nnn2c1CSCC2 C(=O)(CCC(=O)c1cnn(C)c1)N1C(C(N2CCC(C)C2)=O)CC1 c1(C(N2CCC(NC(C(C(C)(C)O)F)=O)CC2)=O)cnc2c(c1)COC2 C1(CNC(C=CSC)=O)CN(C(c2cc(C3(C)CC3)on2)=O)CCC1(C)C c1(OC)ccc(C(O)C(=O)NCC2CCN2C(=O)C=Cc2ccoc2)cc1OC C1(NC(C(C)(C(C)C)NC(=O)OC(C)(C)C)=O)C2CCOC2C12CCCC2 Cc1c(NC2COCC2F)ncnc1N1CC2C(C)C2C1 Cc1cc(CC(=O)NC(C)(CNC(C23CCCC(CO2)C3)=O)C2CC2)cc(F)c1 C(=O)(CCCCNC(=O)CC1CC(=O)NC1=O)NCC1(C(=O)OCC)CC1 C1(NC(Cc2c(C)noc2Cl)=O)CCN(C(C2(C)COC2)=O)CC1(C)C c1(C(C)(C)C)cc(C(=O)NCCC2CC2(Br)Br)n(-c2ccc(F)cc2)n1 C1(C2CCOCC2)(C(=O)NC(CC)CNC(c2ccsc2Cl)=O)CC1(F)F c1(CSC)ccc(CC(N2CCCC2CNC(=O)CC2CC(=O)NC2=O)=O)cc1 c1(-c2onc(C(CC)(C)C)n2)ccc(C(=O)OC)nc1 N1(C(C)=O)CCC2CN(C(=O)CCC(=O)c3ccc(C)cc3)CC2C1 C1(C(=O)N(CC(C)O)CC)(NC(c2nc(CCC)oc2)=O)CCC(C)(C)C1 c1(CCC(=O)NCC=CCNC(C2C(CC)C2)=O)c(F)cccc1F C(=O)(CC(C)(C)C1CC1)NCC(CC)NC(=O)C(O)CF C1(C(=O)NCc2ccc(CNC(c3nc(C)n(C)c3)=O)cc2)CNC(=O)CC1C C1(C)(C(=O)NC)CCN(C(=O)C(Cc2ccoc2)NC(=O)Cc2ccn(C)c2)C1 CC1CCC(CCC(=O)NCc2ccoc2C(=O)NCC2(CF)CCC2)O1 CC1CCN(C(=O)C(C2CCCN(C(=O)CC3CCCC(=O)C3)C2)C)CC1 c1(CC)ccc(O)c(C(N2CCCC2CCCNC(=O)COC(C)C)=O)c1 c1(C(N2CC(F)CC(NC(C(C)CC(N)=O)=O)C2)=O)n[nH]c2c1CCCCC2 c1(OC)ccc(C)cc1OCC(=O)NCC1CN(C(=O)CC(=O)N(C)C)CC1C Cc1cc(=NC2CN(C(=O)C(C)CC(C)(C)C)CC2C)nc(-c2ccncc2)[nH]1 n1(CCOC)nc(CC2CCC2)nc1-c1cnc(C2CCOCC2)o1 C1(C(N(C2CC(C(N3CCCCC(C)(C)C3)=O)C2)C)=O)CC2CC(=O)C1C2 C1(NC(C(C)=CC)=O)CC2(CCC(NC(=O)Cc3csc(C4CC4)n3)CC2)C1 c12cccc(c1)OC(=O)CC2.c1(C(=O)NC(C)CO)ccccc1O C1(CC)(NC(=O)CC2CCCCC2)CCCN(C(=O)CC(C)n2cccn2)C1 c1(OCC(=O)NCCCNC(c2cc(F)c(F)cc2O)=O)ccc2c(c1)CCC2 C1(C#N)(CC(=O)Nc2c(OC)cccc2)CCN(C(=O)NN2CC(C)OC2=O)C1 c1(C(N(CCC)C(C)C)=O)n[nH]c2c1CN(C(C1COC1)=O)CC2 CCC(C(=O)NCCC(C)(C)NC(C1(c2ccnc(Cl)c2)CC1)=O)C(C)C C1(NC(C2(C)CCN(C)CC2)=O)CCN(C(c2cc(O)cs2)=O)CC(C)(C)C1 c1(C(=O)NCC(C2CCC2)NC(CC2C(C)(C)C2)=O)ccc([N+](=O)[O-])cc1 C1(O)(CN(C)C(C2CCC(=O)O2)=O)CCN(C(c2cc(-c3ccco3)on2)=O)C1 N1(C(C2(C)CC(=C)C2)=O)CC2CCN(C(=O)C(O)CCSC)CC2C1 c1(OC)cc(C)cnc1C(=O)NC(C)CC(C)NC(C1CCCOC1C)=O c1(C(C(=O)NCC(C)NC(c2c(C(=O)OC)nn(C)c2)=O)C)ccc(F)c(Cl)c1 N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC2C(N2CC(N3CCCCC3)C2)=O)C1 CC1OC(=O)NC1C(=O)N(CCC(=O)NCCCN1CCC(O)CC1)C N1(C(CCSCC)=O)CC(NC(c2c(Br)ncn2C)=O)CCC1C O(NC(=O)CCNC(=O)C(Cn1cncn1)N(C)C(C)=O)CCCOC.OCC CC(CC(F)(F)F)C(=O)NC(CNC(c1cc2c(=O)[nH]ccn2c1)=O)C1CC1 c1(C(=O)NC23C(n4cc(C(N)=O)nn4)CC(CC2)C3)cccn2nncc12 c1(C(=O)NC2CCC(CNC(C(C(C)C)O)=O)C2)cc(Cl)cc(Cl)c1 C(=O)(C(C)(C)CO)N(CC(CC)NC(C1CC(OC(C)C)C1)=O)C CCC(CC)C(=O)N1CCC(CCOC)(NC(=O)COc2ccc(C)cc2)C1 c1(C(N(CC(CC)NC(=O)C(C(C)C)NC(N)=O)C)=O)ccn2ccsc12 N1(C(c2ccc(NC(C)=O)nc2)=O)CCC2(CCN(C(C3(C4CC4)CC3)=O)C2)C1 C1(N)(CCCC(=O)NC(c2cncn2C)C)CCOCC1 C#CCC(C(=O)NC)C1CC1.c1(C(N2CC(CC=C)(OC)C2)=O)cc(CC)ccn1 c1(C(N)=O)cc(C(N2CC=CC(NC(=O)C(=O)NCC(F)F)C2)=O)ccn1 CC(C)CCCCCC(=O)NC(CC(=O)NC(CO)CCCO)C(C)(C)C c1(C(N2CC(C)CC(NC(CCC(=O)NC)=O)C2)=O)c(C)[nH]cc([N+](=O)[O-])c1=O C(=O)(CC#Cc1ccccc1)NCC(C)Oc1ccccc1 CCC(CCOC)C(=O)N1CCOC(CNC(c2ccc(C(O)CF)cc2)=O)C1 CC(C)C(C(=O)NCCC1CC(NC(c2cc(O)n(C)n2)=O)C1)c1ccn(C)n1 C12(C(N(C(CCNC(CC(C)O)=O)C)C)=O)CCCC1CCC2 CCCC(C)CC(=O)N1CCCC(N(C(c2cn(C)nc2C2CCC2)=O)CC)C1 c1(OC)ncc(C(N2CCC3CCC23CNC(c2cccnn2)=O)=O)cc1Cl c1(NCCN2CC(C)(OC)C2)nc[nH]c(=NCC2CN(C)CCO2)c1C N1(C(CCN(C(Cc2c(C)non2)=O)C2CC2)=O)CCC2CN(C)CC12 N1(C(C(C2CCCC2)OCC)=O)CCN(C(=O)Cn2cc[n+](C)c2)CCC1C C(=O)(C1=CCCC(C)(C)C1)N(CC(CC)NC(=O)CCC1CCCOC1)CC C#Cc1ccnc(C(=O)NCC2CCCCN2C(C23CSCC2C3)=O)c1 C(=O)(C(O)CCN(C(=O)C(C)(CC)SC)C)NCCC#C c1(C(CC)(C)C)ccc(C(=O)NCC(C)CNC(c2cc(C)oc2CC)=O)cc1 CC(C)S(=O)(=O)CC(=O)NCCC1CN(C(C2(S(C)(=O)=O)CC2)=O)CC(C)O1 c1(OCC)cc(C)c(-c2ccnc(NCc3ccc(O)cc3C#N)c2)cc1C c1(CNC(CC(CONC(c2c(COC)cnn2C)=O)C)=O)ccc(Cl)c(F)c1 C1(C(N(C(C)CNC(=O)C(F)n2cccn2)CC)=O)CCC(C(=O)OC)C1 c1(OC)ccc(CCC(N2CC3CC2(CNC(=O)C2=CCCC2)C3)=O)c(F)c1 N1(C(C(CC)O)=O)CCN(C2CCN(C(=O)CS(=O)(=O)NC3CC3)CC2)CC1 O=c1c2ccccc2nc(-c2ccccc2)n1CC1C2COCC12 N1(C(C2(CCC=C)CC2)=O)CCC(O)(CN(C)C(C2CCCCC(=O)N2)=O)CC1 C(C)(C)(CC(F)C(=O)NC(c1ncc(C)cn1)C)NC(c1cc(CC)no1)=O C1(NC(=O)C=Cc2nccs2)CN(C(C2CCS(=O)(=O)N2)=O)CC2(CCC2)C1 N1(C(C(CCC)C)=O)CCC(C2CCCN(C(=O)C(c3c(C)noc3C)C)C2)C1 c1(C(=O)NCC2CCCN(C(CCC(=C)C)=O)CC2)nccc2c[nH]nc12 C1(CNC(c2ccccc2NC)=O)COCCN(C(c2ccc([N+](=O)[O-])o2)=O)C1 CC(CC(=O)NCC1(CCNC(=O)Cn2cccn2)CC1)C(F)F Cc1nn(C)cc1C(=O)NCc1ccc(CN(C)C(C2CCCNC2=O)=O)cc1 c1(CNC(C=CSC)=O)nn(C)c2c1CN(C(=O)CN1CCS(=O)CC1)CC2 c1(C(N2CCCC(O)(CNC(C(C(C)C)OCC)=O)C2)=O)ccc2c(c1)OCC2 C1(C(=O)NCC(CCC)CCO)CC2CCC(C1)N2C(=O)CCCNC(C)=O CCCCCCCCCCC(c1nnnn1C(C)C)NC1CCCC1(C)C N1(C(=O)NC(c2ccncn2)C)CCOCC1Cc1ccc(Br)cc1 C12(NC(c3c(N)non3)=O)COC(C1)C(NC(C1CC3CCC1C3)=O)C2 c1(CN2CC(C(=O)Nc3c(OC)nc(C)nc3)C2)ccc2ccc(O)cc2c1 CC1(C)CCC(C)(C)N(c2ccnc(NCCCc3cn[nH]c3)n2)C1 C=CC1(C(=O)NCc2nccc(C)c2F)CCN(C(C2C3COCC23)=O)CC1 C(=O)(C1=C(Cl)CCCC1)NCCCNC(C(c1cccc(Br)c1)(C)C)=O Cc1cc2c(=O)c(C(=O)NC3COCC3NC(=O)C=CBr)c[nH]c2[nH]1 C1(NC(=O)CC2(Cc3ccon3)CC2)CC2CCC(C1F)N2C(=O)C(O)C1CC1 C12CN(CC1O)CCOCCC(=O)NC2.c1(N)ccnc(Cl)n1.CO C1(CNC(CCn2ccc(C)n2)=O)CCCC(NC(=O)CC(C)(F)F)C1 C(CC(C)C)(C(=O)NC1CC(C)(CNC(C2CCC(=O)N(C)C2)=O)C1)NC(C)=O C(=O)(CC(C)N1CCCC1=O)N(CC(CC)NC(CCOCCC)=O)C C1(NC(C2(SC)CC2)=O)CC2(CCN(C(C3CCC(CC(=O)OC)O3)=O)CC2)C1 C(=O)(CC(CC(C)C)NC(=O)CC1(O)CCOCC1)NC1(CCC)CC1 C(C(C(C)C(C)C)NC(c1ccc(N)c(Cl)c1)=O)NC(c1c(C)scc1)=O Cc1onc(C(=O)NC(CNC(c2cc3n(n2)CCC3)=O)CO)c1[N+](=O)[O-] CCC(CC)C(C(=O)NCC1(CNC(=O)CC(C)C(=O)OC)CCC1)OC C(=O)(CC(C)C(=O)NCCC1CCCN(C(=O)C(C)(C)c2cncs2)C1)OC CC(C)C(O)C(C)C(=O)N1CC(O)CC1CNC(C12CCCC1C2(F)F)=O C1(NC(C2(N(C(COCC#C)=O)C3CC3)CCC2)=O)(CSC)CCOC1 C12(C(N(C)CC3CCN(C(c4nsnc4O)=O)C3)=O)CCC(CC1O)C2 c1(C(C)OC)cn(C2CN(C(c3cc(Br)no3)=O)C2)nn1 N1(C(C(CCOC)C)=O)C2CCC1CC(C(=O)NC1CCCN(C(C)=O)C1)C2 N1(C(C2(OC(C)=O)CC2)=O)CC(C)(NC(c2cnc(O)o2)=O)C1 c1(CC=C)cccc(C(N2CCC(C)(C(=O)NC(C)C(C)n3cccn3)C2)=O)c1 CCC(O)C(C)C(=O)NCCC(CNC(=O)CCc1nccn1CC)OC C(=O)(C(C)CC(F)(F)F)NCC1CN(C(c2cc(C)c(C)nc2)=O)CC1(C)C C=CCC(CC)C(=O)N1CC(OC)C(NC(=O)CCOC2CCCCCC2)C1 C1(Cl)(C(=O)NCC(CN(C(C2CCC(=O)N2)=O)CC)(C)C)CC12CCC2 c1(C(=O)NC2C(OC)CN(C(C3(F)CC3C)=O)C2)csc2ccc(F)cc12 C1(CC=C)(C(=O)NCC2(CO)CC=CC2)CN(C(c2ccn(C)c2)=O)C1 c1(OC)cccc2c1CC(Nc1ncc(S(C)(=O)=O)cn1)C2 N1(C(=O)C(O)C2CCC2)CC2(CCCCN2C(c2cnc(C3CC3)[nH]2)=O)C1 Cc1c(CNC(N2CCN(c3ncc4ccccn34)CC2)=O)sc2nccn12 C1(NC(C2(CCC)CC2)=O)CCCCN(C(=O)CCn2ccnn2)C1 c1(C(=O)OC)ccc(NC(C2CN(Cc3cccc(I)c3F)C2)=O)c(Cl)c1 c1(CC)occ(C)c1C(=O)NCC1CC1NC(=O)C(C1CC1)C1CC1 O=C(CCCCCF)NCC1CCC1NC(=O)Cn1nnc(-c2ccccc2)n1 N1(C(c2ccc(-c3nn[nH]n3)o2)=O)CC(O)CC1c1cn(-c2nccs2)nn1 N1(C(C(CC)(C)CO)=O)CCCN(C(=O)CCOCCC(=O)OC)CCC1 CC12CN(C(=O)COCCF)CC1CN(C(c1nnn3c1CCCC3)=O)C2 C1(NC(C2CC(NC(C3CC3C3CC3)=O)C(O)C2)=O)CCC2(CCC2)CC1 C(N=c1cc(NCCC2CC3CSCC3C2)nc(C(F)(F)F)[nH]1)c1ccc(C)cc1 N1(C(C(COC)O)=O)CCC2(CCN(C(=O)CC3CN(C)C3)CC2)C1 Cn1ccc2c(C(N3CC(NC(=O)CCN4CCCC4)C(C)(C)C3)=O)cccc12 c1(C(=O)NC(CC2CN(C(c3cccc(C)c3N)=O)C2)C)ccc2nn[nH]c2c1 c1(CNC(=O)NC2CC3CCC2C3)ccc(C(F)(F)F)c(F)c1 c1(CC)ncc(C(=O)N(C2CN(C(=O)C(C)(C)c3cnco3)CC2F)C)c(O)n1 c1(C(=O)NCC(C)CN(C)C(C2C3CCCC23)=O)cccc(CN(C)C)c1 C=Cn1ncc(C(N2CC3(C(=O)NC4CCSC4)CC2CO3)=O)c1N C(=O)(CCC(C)S(C)(=O)=O)N1C2CC(CNC(CSCC)=O)CC1CC2 c1(C(=O)NCC2N(C(C(CC)COC)=O)CCC2)nc(Cl)ccc1Cl CCC(C)(COC)C(=O)N1CC(N(C)C)C(C(F)F)C1.C12(CCC1)C(=O)NC2 Cc1c(N)ccc(C(=O)NC2CN(C(=O)CC3C=CCC3)CC2CC2CC2)c1C c1(C(C(=O)NC2CCOC2)N(C)Cc2cc(C3CC3)on2)ccsc1COC C(CC(O)CCc1ccccc1)NC(Cc1onc(C)n1)C Cc1ccc2snc(C(N3CCC(C)C(CNC(=O)CCC(C)C)C3)=O)c2c1 Cn1cc(Cl)c(CC(=O)NCC2C3CN(C(=O)COc4cccnc4Cl)CC23)n1 S(=O)(=O)(C(C)CC(=O)Nc1ccccc1N(C)C)N(c1cccc(Cl)c1Cl)C C1(CC(=O)NCC(C2CCC2)OC)COCC1NC(=O)CCn1cccc1 n1(CC)nc(C)c(C(N2CCC(O)(C(C)NC(=O)Cn3nnc(C)n3)C2)=O)c1Cl c1(C(=O)NC2(CNC(C(=Cc3cccnc3)C)=O)CCC2)cc(N)cc(O)c1F CC1CN(C(=O)C(=O)NC2CCOCC2)CCN1C(C12COC(C1)C2)=O C1(C(N2CCC(CC(=O)N(C(C3(C)CC3)C)C)C2)=O)CC(=O)CC(=O)N1 c1(C(N2C3CC(CNC(C(CC=C)C)=O)C2CC3)=O)ccc(S(N)(=O)=O)c(C)c1 CC1(C)CC1(C(=O)NCCC(F)(F)F)NC(=O)CC1C=CCC1 C=C1C(C(=O)N(C(C)C(=O)NCC(C)C2CCC2)C)C1C(=O)OC C1(CNC(C(C(C)C)CN(C)C)=O)CCCC2CN(C(c3cnnn3C)=O)CC12 c1(C2(C(=O)NCC(C)NC(c3nccc(C(F)F)n3)=O)CCC2)cccc(Cl)c1 C1(NC(C2CCC(C)C2)=O)CN(C(=O)CCC(C)(F)F)CC(C)(C)C1 N1(C(C2(OC)CCN(C(C3OC4CCC3C4)=O)C2)=O)CCc2ccncc2C1 c1(C(=O)NCC(C(C(=O)NCC(CC)CC)F)C)cnc2ccccn12 CCCC(C)(CC)NC(=O)CC1CCCCC1NC(=O)CSC(C)C c1(CN(C(=O)CCNC2(C#N)CC2C(F)(F)F)C)ccccc1Cl N1(C(CCC=C)=O)CC(OC)CC1(C)CNC(=O)COCC(C)C C(CC(=O)NCCCCCCO)(C(C)C)NC(C(C)N(C)C)=O c1(CC(N2CC(C=C)C(NC(=O)C(CO)C(C)C)C2)=O)ccc2c(c1)CCCC2 C(=O)(C(C#N)C(C)(C)C)NCC(C)C(N1CCC(C2CCC2)C1)=O Cn1c(=O)oc2cc(CNC(=O)CCCCCn3cc(CNC)nn3)ccc12 CCN=c1[nH]c(C(=O)NCC2CCCC(CNC(=O)CN3CCC(C)C3)C2)cs1 c1(OC)cc(OC)nc(N2CCC3C(OC)CC23)n1.c12ccc(cc1)c(=O)[nH]2 N1(C(C(CC(C)C)NC(C)=O)=O)CCC2(CC1)CC(NC(C1(C#N)CC1)=O)CCO2 C(=O)(C(C(C)CCC)N(CC(=C)C)C)NCC(=C)C c1(C(=O)NC2CC(NC(CSc3n[nH]c(=N)s3)=O)C2)cc2cc(Cl)ccc2s1 C1(CC(=O)NC(COC)C2(C)CC2)CCCCN1C(=O)CCc1cc(C)[nH]n1 CC1C(C(=O)N(C)CCOCCNC(c2ccnn2CC(F)F)=O)CCN1C c1(C(=O)NCC(C2CC2)NC(c2c(OC)cc(C)cc2)=O)nc[nH]c2nccc1-2 C1(CNC(CCC#C)=O)CCCC(CNC(c2cccc(C3CC3)c2)=O)C1 c1(C(N2CCC(C(C(C)C)NC(C#CC(C)C)=O)CC2)=O)nc(O)nc(O)c1F N1(C(C)(C)C)CCCCCC1c1ccco1.C12CC(C(O)C1)NC(=O)N2 C12(NC(c3cnc(COC)s3)=O)CCN(C(C3(COC)CCCCC3)=O)CC1C2 C1(CNC(c2cncc(SCC)n2)=O)CCN(C(C2CC2(C)C)=O)CCC1(F)F C1(C(N2CC3C(CNC(C(C)(C)OC)=O)(C3)C2)=O)CC2OC(=O)OC2C1 c1(C(=O)NC2CC(NC(C3C(OC)CCCC3)=O)C2)n[nH]c2c1CCCC2 C(=O)(C(Cc1cccc(C)c1)CC)NCC1C(NC(c2ccn(CCC)n2)=O)C1 c1(CN(C(=O)CC2(C(F)F)CC2)CC2CC(C(=O)OC)C2)ccccc1 N1(Cc2cc(C(F)(F)F)cc(O)n2)CCCCC1C1(C(F)(F)F)N=N1 c1(CNC(CC=C=C)=O)cc2n(n1)CCN(C(=O)C=Cc1cnc[nH]1)C2 c1(C(=O)NCC(N2CCN(C(C=CCCC)=O)CC2)=O)cc(C2CC2)cnc1O CCCCC(O)CC(=O)N1CCC2(CC1)CC2CNC(c1cc(OC)ncn1)=O C12(NC(=O)C(F)=C3CCCC3)CC(C1)N(C(=O)CCOc1cccc(Cl)c1)C2 N(C1CCn2nncc21)C1(c2cn(C(C)C(=O)N(C)C)nn2)CCOCC1 C(=O)(CCCC(CC)NC(C1C2CCC(F)C12)=O)N(C)CC N1(C(c2ccc(C)n2C)=O)CCC12CN(C(C1(C)CC1(F)Cl)=O)C2 c1(C(N(C2CCN(C(=O)C(c3cnn(C)c3)OC)CC2)CC)=O)cccc(=O)o1 C12C3CC1N(C(=O)Nn1cccn1)C3C(O)CCC(=O)O2.c1(C)ccccc1 C(CC(C)C(C)(C)C)NC(c1c(C)oc(CNC(=O)CC=CC(C)(C)C)n1)=O N(C(=NCCCOCC)NCC1CCCC1O)CCCCCC S(=O)(=O)(c1c(C)noc1C)N1CCN(C(CC(=O)OC)=O)CC1C(F)(F)F c1(CNC2C(C(=O)NC3CCCCC3)C2)cccc2ccoc12 C(CCC(=O)N(CC(O)CO)C)N(C(C)C)C.C12(CC1)CC(=O)N2 c1(C(C)=O)cc([N+](=O)[O-])ccc1N1CCC(NC(=O)C(C)(C)C2CCC2)C(O)C1 Cc1cc(-c2nc(-c3cnn(C)c3)nn2C(C)C(C)C)cc(=O)n1C C1(C(=O)NCC(CO)OC)(SC)CCN(C)C1 c1(OCCC)cccnc1C(=O)NCC(C)CN(C(=O)C1=CCSC1)C C1(NC(C2CC23CCC3)=O)CC(O)C1CC(=O)NC1COCC1C(N)=O c1(NC(C(c2cnn(C)c2)NC(C(CC)n2ccnc2)=O)=O)ccc(O)c(C)c1 C1(CNC(CSC)=O)CC2(CCN(C(C3CC3C3CCCO3)=O)CC2)C1 N1(C(Cc2c(C)scc2)=O)CC(O)CC1(C)C(=O)NC(c1nnnn1C)C c1(CC(=O)N(CCCCCC(=O)NC(=O)C(O)C2CC2)C2CC2)sccc1Br N1(C(c2cnn3ccc(C)cc32)=O)CCC2CN(C(=O)CN(C)C(C)C)CC2C1 N(C1CCCn2cnnc21)C(CCCCCNC(=O)Cc1cccnc1)=O c1(C(N2CCCCC2c2nc[nH]n2)C(=O)NC2CCOC2)ncccc1F C1(CNC(C(C)(F)F)=O)CCCC(NC(=O)CCNC(C2CCOCC2)=O)C1 C1(C(N2CCOC(C(N)=O)C2)=O)CC(F)CN1C(c1ccn(CCF)n1)=O N1(C(c2cnc(C(F)(F)F)nc2)=O)CCC2CN(C(c3ccc[n+]([O-])c3)=O)C2C1 C1(CNC(c2scnc2Cl)=O)CC2CCC1N(C(c1c[nH]c(Br)c1)=O)C2 c1(OC)ccccc1C=CC(=O)NC(C)CC(C)NC(=O)Cc1cncc(O)c1 n1(CC(C2CCOCC2)CO)cc(-c2cc(C3CCCO3)n[nH]2)nn1 N1(C(C2CCOCC2)=O)CCC(NC(C2(n3cc(Br)cn3)CC2)=O)CC1 N1(C(C2(C)C(C)(C)C2)=O)CCC2(CC1)CN(C(c1ccccc1Cl)=O)CCO2 N1(C(C2N(C(C3CNC(=O)N3)=O)CC(O)C2)=O)CCC(O)CC12CC2 c1(C(N2CCC(n3cc(CCNC(N)=O)nn3)C2)=O)coc2c1NC(=O)CCC2 CC1=CCC=CC1C(N1C2CCC1CC2)=O.c12cccc(c1)C2 C(Cn1cncn1)(C(=O)NCCN1CCOC1=O)NC(C(C)NC(N)=O)=O c1(C(=O)NC2CN(C(c3cc(C)c(F)cc3)=O)CC2O)cc2cncn2c(O)n1 O(N=C1CCCCCC1)CC(N1C(CNC(C2(CF)CCC2)=O)CC2CC12)=O c1(OC)cc(C(=O)O)ccc1CNC(c1ccc(Cl)cc1)C(F)F S(=O)(=O)(c1ccccc1Cl)NCC(=O)Nc1c(CCCOC)c2c(s1)cccc2 C1(C(=O)NC2(CN(C(C(CC3CC3)OC)=O)C)CC2)Cc2nccn2C1 N1(C(c2nn(CC)c(C)c2)=O)CCC(NC(=O)CC2CCCC(F)(F)C2)C(F)C1 C1(CNC(c2cc(CCO)on2)=O)CN(C(c2cn(C(F)F)cn2)=O)CCCO1 C(=O)(C(C)CC(C)(C)C)NC(C(=O)NCCCCCC=C)CN=[N+]=[N-] N1(c2c(OC)cncn2)CCC(C)(C)C(CNC(=O)C(C)(C)N2CCOCC2)C1 N1(C(C(CCC)OCC)=O)CC(=O)NCC1C(=O)NC1CCCCC12CC2 c1(C(=O)NCC(CN(C)C(C2(Cl)C3CCC(=O)C23)=O)O)cnc2occc2c1 CC1(C)CC(NC(=O)CC2CC(F)(F)C2)CN(c2cc(O)ncn2)C1 C=CC1CCCCN(C(=O)Cc2cccc(Cl)c2OC)C1 N1(C(c2cccc(C)c2N)=O)CCC(NC(=O)CC(C)N(C)C)C(C)(C)C1 C12(NC(CCCNC(=O)OC)=O)CCCC1(F)CN(C(=O)COC(F)F)C2 C1(NC(CC=C)=O)CCCC(Nc2c(NC(=O)Cn3ccnn3)cccc2)C1 N1(C(C(c2cccc(C)n2)NC(C(C=C)C)=O)=O)CC2C(C1)C2(C)C C1(CC(=O)NCC2CC(NC(C3(CC=C)CCOC3)=O)C2)CCOC1(C)C c1(C(=O)NC2CCC(CNC(CN(C(C(C)C)=O)C)=O)C2)ccc2cc(C)cn2c1 c1(C(=O)NC2C=CCN(C(CCC=C(C)C)=O)C2)cncc2nc[nH]c12 CCC(CC)C(C)C(=O)N(CC(O)CNC(c1ncc(C(=O)OC)cc1N)=O)C C1(C(=O)NCC(=O)N(C)CC)C2CC3C(C2NC(=O)CC2(O)CCC2)C13 N1(C(c2cccc(NC(CC)=O)c2)=O)CCCOC(CNC(c2ccsn2)=O)C1 CC1CN(C(=O)CCCN2CCCCC2)CCC1CNC(=O)CCF c1(C(=O)NCCCC(C)NC(C2(CC)CCC(O)CC2)=O)cc(F)cc(C)c1N C=CCC(CNC(=O)C(C)(C)CCC)C(=O)NCCCC1CCOC1=O C1(C(N2CC3CC(NC(CC4CCC(C)(O)CC4)=O)C3C2)=O)CCCN2CCCC12 c1(-c2ccc(OC)nc2)cnn2c1CN(C(=O)C(C)Cc1ccccn1)CC2 C(C)(C)(CCC(=O)NC1CCCN(C(C)C)C1)NC(c1cncc(OC)c1)=O N1(CCCN2CCCC(O)(c3cc[nH]n3)C2)Cc2cccnc2C1 C#Cc1ccc(C(=O)NCC2(C)CCCN(C(=O)C3=CCOC3)C2)cc1F C1(CCOC)(NC(=O)C2=CCCS2)CCN(C(=O)C(F)C2CCC2)C1 c1(C(=O)NC(C2N(C(c3cc(CC)no3)=O)CCC2)C)cn(C)nc1C1CC1 C(=O)(C(F)C(F)(F)F)NCC(CNC(c1c(CC)n(C2CCCC2)nc1)=O)(C)O N1(C(=O)CC2CC(O)C23CCC3)CC(C2CCN(C(C34CC(F)(C3)C4)=O)CC2)C1 C1(C(=O)O)C2CCC(C2)C1C(N1CCCC(c2ncccn2)C1)=O Cc1occc(=O)c1OCC(=O)NCC(C(C)(C)C)NC(=O)C1=COCCO1 C1(NC(c2ccnn2C2CC2(F)F)=O)C=CCN(C(c2csc(Cl)c2)=O)C1 CCCCC(C(=O)NC(C1CCCN1C(=O)C=Cc1csnc1C)C)NC(N)=O c1(C(=O)NC2C(CNC(CC(CC)SC)=O)CC2)cccc2nccnc12 N1(C(CC(C)C)=O)C2CCCC1CN(C(=O)C(F)(F)CC1CC1)CC2 c1(OC)c(Cl)cc(C(N2CCC(CNC(c3occc3F)=O)C2)=O)nc1Cl C1(NC(=O)Cc2ccoc2)CCCOC12CCN(C(C1CC13CCCC3)=O)CC2 N1(C(C2CN(CC(C)C)C2)=O)CCCCC1CN1CCCC1=O C(=O)(CCCS(C)(=O)=O)NCC1C(C)CCN1C(=O)CCC(=O)c1cccs1 C#CCC(C)(C)C(c1nnnn1CCC1(C)CC1)NC(C)Cc1ccc(Br)cc1 c1(NC(C(=O)NCCCC(=O)N(C)C)=O)cnn2cccnc12 N1(C(C(CNC(C2CCC(=C)CC2)=O)CC(C)C)=O)CCC2(CC1)CC2C#N C1(C(=O)NC2(CC)CCN(C(=O)C(C3CC3)OC)CC2)CCOC2(CCCC2)C1 CCC(CN(C)C)C(=O)N1CCC(OCCCNC(C2(O)CCOCC2)=O)CC1 c1(CNCC2CCN(C(C3CC3F)=O)C2)ccc(-c2ccsc2)cc1 c1(C(=O)NC2CC(NC(c3nc(C(C)OC)oc3)=O)C2)ccc2c(c1)CCCC2 C1(COC)CCN(C(=O)CCn2cc(CC3(OC)CC(=O)N3)nn2)CC1 CCCCCCCCC(=O)N1CC2C(C(N3CCOCC34CCC4)=O)C2C1 N1(C(CCC(C)OCC)=O)CC2CCC(C(=O)N(C3CCCC3)CCO)(C2)C1 c1(C(=O)NC2C(NC(c3n(C)ccn3)=O)CCCC2)sc2ccccc2c1Cl C1(NC(C(COC)N(C)C)=O)CC2CC1CN(C(C1CCC3(CC1)CC3)=O)C2 N(C1CCCc2cccnc21)C(C1CCC(NC(CNC(CCC)=O)=O)CC1)=O c1(C(N(C(C(C)C)C(=O)O)C2CCS(=O)(=O)C2)=O)ccc2c(c1)OCO2 C(=O)(C#CC(C)(C)CNC(=O)CCCC(=O)N(C)C)N(CCCOCC)C N1(C(C=C(C)C(F)F)=O)CCN(C(=O)CN2CCN(C)CC2)C2COCC12 c1(C(=O)NC(C(=O)N2CCC(SC)C2)CN=[N+]=[N-])c[nH]c2cccnc12 c1(OC)cc(CO)ccc1C(=O)NC(C)(C)CCNC(c1ccc(C2CC2)s1)=O CCCCCCC(C)CC(=O)NCCNC(c1ccc(OC)c(N)c1F)=O C(N=c1ccc(S(=O)(=O)NC2CCCC(C)(C)C2)c[nH]1)c1cncc(OC)n1 N1(C(c2ccc(C(=O)OC)s2)=O)C(CNC(C2(C)CC2C)=O)CC2CCCCC12 N1(C(c2cc(C#N)sc2)=O)CCN(C(=O)Cc2cccc(F)c2)C2CC12 N1(C(c2ncc(C(=O)OC)nc2)C(=O)NCCSC)CC(C(N)=O)OCC1(C)C CCC(CC(F)(F)F)NC(C1(NC(=O)CCOC(C)=O)CCN(C)C1)=O C1(C(=O)NC(C2CCN(C(c3cc(C)nn3C)=O)CC2)C)CC2(CCCCC2)C1 CC1CCCC=C1C(=O)N(C(C)(C(N1CC[Si](C)(C)C1)=O)C1CC1)C N1(C(C)=O)CCC2(CC1)CC2(C)C(N1CCCC(O)(CN)CC1)=O CCCCCCC(C)(C)C(=O)NC1CN(C(c2ccnn2CCOC)=O)CC1O C1(C(=O)NCCN(CCC)Cc2ccccc2Cl)C2Cc3ccccc3C12 c1(C(=O)NCCOCCN(C(=O)C(F)C(F)(F)F)C)cn2c(n1)CCC2 C1(CC(=O)N(CCC(=O)OC)C)(COC)CCCC1.C1CC(=O)NCCCO1 c1(OC)ccc(OC)c(NC(=O)NCCCCCc2cnn[nH]2)c1OC C1(CC)C(=O)N(C)CCN1C(c1cnc(Cl)s1)C(=O)Nc1ccccc1Cl N1(C(=O)C(c2ccc(Br)cc2)O)CCCC2(CCCN(S(=O)(=O)CCCl)C2)C1 c1(C(COCC(=O)N(CC(CC)NC(c2ccc(C)s2)=O)CC)C)ccccc1 CC(C)C(C(=O)NC1CN(C(C2C3(CC3)C23CC3)=O)CC1C(F)F)NC(N)=O C1(C(=O)NC2CCCC2(C)CN(C(=O)C(C)(C)C)C)(COC)CCOCC1 c1(C(N(C)CCNC(c2cn(CC(F)(F)F)nn2)=O)=O)cc(C(F)F)cc(F)c1 c1(C(N2C(C(=O)NCCn3cnnc3)CCC2C2CC2)=O)cccc(O)c1 c1(OC)ccc(OCC(=O)NCC2COCCO2)c(Br)c1 C(=O)(C(CO)C(F)(F)F)NCCCC1N(C(CCc2cn(C)nn2)=O)CCCC1 N1(C(CCC(CC)C)=O)CC(C(=O)NCC2(CC)CC2)C2(CCC2)C1 n1(CC)sc2ccccc2c1=O.n1(COCCO)nc(C)c(C2(CC)CC2)c1C N1(C(C(C)NC(CC)=O)=O)CCN(C(=O)COc2ccc(C)cc2C)CC1CO c1(C(=O)NCc2cc(C(N(CCOCC#C)C)=O)no2)ccnc(CC)c1 c1(COCC)nnc(CNC(COC(c2cc(Br)c(Br)s2)=O)=O)n1C N1(N2C(=O)CN(C(=O)OC(C)(C)C)C2CC)CCS(=O)(=O)C2(CCCC2)C1 N12CC(C(=O)O)C3(C1)CN(C3)CC2=O.C1(C)(C(N2C(C)CCC2)=O)C=CCCC1 C1(C#CC(=O)NC2CC3C(NC(=O)CCC(C)C)C3C2)(CC)COC1 C(=O)(C(C)CCCc1ccccc1)N1CCCC(N(C(c2cnns2)=O)CC)C1 N1(C(c2cncn(C)c2=O)=O)CC2CN(C(c3ccccc3Cl)=O)CC2(C)C1 c1(C(=O)NC(C(C)NC(c2c(SC)scc2)=O)C)cccc(C#N)c1 C=CC(C)(O)CC(=O)N1CCC(NC(=O)COc2ccc(C)cc2C)CC1 c1(C(=O)NC2(C(=O)NC3CC(N(C)C)C3)CC2)cnccn1 CC1CN(C(C2(C)CCNC2=O)=O)CCC1CNC(C1CCOC1)=O N1(C(C(C2CC2)SC)=O)CCCCC1c1ccc(C(=O)NCCC2CC2)n1C N1(CC)CCOCC1CC(=O)OC.C1=CC(=O)NC(C2CCOC2)CNC(=O)C1 C12(NC(CCC=C)=O)CCC(CC1NC(c1cc(C(C)C)no1)=O)C2 CC(C)(C(=O)N1CC2CC(NC(c3csc(-c4ccsc4)n3)=O)C1C2)C(N)=O c1(OC)cc(CN2CCN(C(c3coc(C(C)C)n3)=O)CC2)cc(OC)c1OC n1(CCC)nc(C)c(C(=O)NC2CS(=O)(=O)CC2NC(c2ccco2)=O)c1C c12cn(nn1)CC(=O)N(C)C2c1ccncc1.C1(CCC)(C(=O)OC)CCC1 CC1(CNC(c2ccc(Br)cc2)=O)CCCN(C(C2COC(=O)C2)=O)C1 C1(CNC(CCN(C(C(C)n2cccc2)=O)C)=O)CCC(CO)O1 n1(CC(N2C3CC(NC(c4c(OC)c(Cl)sc4)=O)(C3)C2)=O)ccc(C)cc1=O c1(C(N(CCC)CCNC(=O)C(CC)N(C)C)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(=O)N(C23CC(C2)C3)C(C2CC2F)=O)c(C(F)(F)F)nc2ccccn12 C1(CC(=O)NC2CN(C(CC)=O)C2)CCCCN1C(C1CC(C)=NO1)=O c1(C(N(CC(CNC(C(CC)OCC)=O)C)C)=O)cnc2n(c1=O)CCS2 N1(C(C(c2ccc(C)s2)C)=O)C2CCC1CC(CNC(=O)Cc1sccc1C)C2 N1(C(c2cc(C)n(C)c2)=O)CCCC(C)(CNC(C2(O)COC2)=O)C1 c1(OC)cc(Cl)ccc1C(=O)NC1CC(C(C)NC(C2CC=CC2)=O)C1 c1(NC)cc(C(F)(F)F)nc(CNC(N2CCNC(=O)C2c2cnn(C)c2)=O)n1 CC1CC2(CC2)CN1C(C1C(NC(c2c[nH]nc2Cl)=O)C1(C)C)=O c1(C(=O)NC(C2(O)CN(C(CCOC(CC(C)C)C)=O)C2)C)ccc(Cl)c(F)c1 CCC(CC(=O)N1CCC(CNC(c2nnc(O)cc2O)=O)CC1)C(C)(C)C c1(C(N2CCC(C3CC3)C2)C(=O)NC(C)(C)C)ncc2ccccn12 C1(C(=O)NC(CC=C)C2CC2)CC(C)CN(C(=O)CC2CCN(C)CC2)C1 Cc1cccc(NC(=O)C(c2cn(C)nn2)NC(C2COCOC2)=O)c1 c1(CNC(C2(F)CN(C(=O)C(F)F)C2)=O)ccc(Br)cc1.C(c1ccco1)=C C1(C(N2CCC(C(=O)NC3(CO)CCCCCC3)CC2)=O)CS(=O)(=O)CC12CC2 Cc1ccc(CNC2CN(C(c3cnc(C)s3)=O)CC2F)c(C)c1 C1(CC(=O)NCC2(CNC(C(OC)OC)=O)CC23CCC3)NC(=O)CNC1=O c1(C(=O)NCC(CCOC)NC(=O)CNC(c2cn[nH]c2)=O)ccncc1F C1(C(N2CCC(NC(c3cc(O)ncn3)=O)C2)=O)Cc2cccnc2C1 N1(C(C(CC)(C)COC)=O)CC2CCCN(C(c3n[nH]c(C)c3C)=O)C2C1 n1(CC(=O)NCC2CN(C(Cc3c(C)non3)=O)C(C)C2)cc(Br)ccc1=O N1(NC(C)C)CC(=O)N2CCCC2C1.N12CC(COC1=O)SC(C)C2=O c1(CN2CC3CN(C(C(c4c(C)cc(N)cc4)=O)=O)C3C2)cn2ccccc2n1 c1(N2CC(C(C)NC(CSCC#C)=O)OCC2)ncnc2cc(C(C)C)nn12 c1(C(N(C)CC2CN(C(C3C=CCC3)=O)CCO2)=O)cccc2nc(CO)[nH]c12 C12(C(N(CCCOCC)C)=O)CCC(CN(C(c3ncncc3OC)=O)C1)C2 C=C1CCC(C(=O)NC2CC2CNC(c2nc(C)n(C)n2)=O)CC1 N1(C(c2cc(OCC)n[nH]2)=O)CCN(C(C2C3CNC(=O)C23)=O)C2COCC12 C(=O)(C1=NNC(=O)CC1)N(C1CN(C(C2CCC(C)(C)CO2)=O)C1)C c1(C(=O)NC2C3(CC(NC(c4cc(=N)[nH]cc4)=O)C3)C2)cc(F)cc(F)c1 C1(CC=C)(NC(C)=O)CCN(C(=O)C(CC)NC(=O)CN2CCCC2=O)C1 c1(C(=O)NC(C2CCN(C(=O)C(C3CC3)N(C)C)CC2)C)ccc(CCF)cc1 C(=O)(C#CC1CCCO1)NCC1(NC(C(c2c(C)n[nH]c2C)C)=O)CC1 N1(C(C2C(C(=O)OCC)CC2)=O)CCCCC(NC(C2CCN(C)CC2)=O)C1 CCCC(C(O)C(=O)NC1CCCCCC1C)NC(=O)C(C)CC(C)(C)C c1(Nc2nc(NCC3C(C)CCC3)c3c(n2)scc3)ncc2ccc(Br)cc2n1 C(=O)(CC(C)(C)C(F)F)NCC(CC(=O)NCc1nccc(C)n1)(C)C C12(OC)CCC(C(=O)NCCC3CN(C(c4cnc(C)n4C)=O)CCO3)(CC1)C2 c1(C(N2CC(OCC=CCC3CCCN(CCF)C3)C2)=O)noc(C)c1C=O.CO N1(C(C2(COC)N(C(CCC)=O)CC=C2)=O)CCCOC(COC)C1 c1(C(c2n(CCC)nnn2)NCc2sc(C)nc2C)cc2ncc(Br)cc2o1 c1(C(ONC(=O)NCC2CCN(c3ccncc3)C2)C)cnn(C)c1F C1(NC(c2c(CCC)nns2)=O)CN(C(C2CC(=O)NC(C)C2)=O)CC12CCC2 Cc1occc(=O)c1OCC(=O)NCC(CC(C)C)NC(C1(C)CC1Br)=O C1(NC(CCCNC(c2cc(C)[nH]c2C)=O)=O)CCC2CCCC1O2 N1(C(c2c(OC)cccn2)=O)CCCC2(C1)CN(C(c1cc(Cl)no1)=O)CCO2 C1(NC(Cc2cc(CC)on2)=O)CS(=O)(=O)N(C)C1(C)C Cc1cc(C(=O)N(C2CN(C(c3ccnn(C)c3=O)=O)CC2F)C)c(C)cc1Cl c1(CCC(=O)NCCC(F)Cn2cc(C3CCCC3)nn2)ccc(F)cc1 C#Cc1ccc(CC(N2CC(OC)CC2Cc2cccs2)=O)c(Br)c1 n1(CC(N2C3CC(NC(C4CC(N(C)C)C4)=O)C2CC3)=O)ccc2ccccc12 c1(C(N(CCC(=O)NCCN2CC=CC2)CC#C)=O)cc(C)c(C)s1 C12(C(=O)NCC(C)(CO)NC(c3nn(CC)c(C)c3)=O)CCC(C1)C(C)(C)O2 C1(C(=O)OC)CCOC1C(=O)NC1CC(CCC(=O)N(C)CC2(SC)CC2)C1 c1(C(N2C(C(=O)NC(CC)(C)C)CC(O)C2)=O)ccc(OC)cc1OC1CC1 CC(CC(=O)N(C)CC1CCC(NC(=O)CN(C2CCCC2)C)CC1)C(F)F C1(CCN(C)C(c2cncc(Br)c2)=O)CCN(C(=O)C(c2ccccc2)F)CC1 CC(C)(C(=O)O)n1cc(CCC(c2ccccc2)O)nn1.C1(=O)CN1 C(C1CCCN1C)=CC(NOCC(=O)NC(C)CF)=O C(=O)(C1c2ccccc2C2CC1C2)NCC1(N(C(CCSCCCC)=O)C)CC1 C1(NC(Cc2n(CC)cnn2)=O)CCCC(N=c2cc(C)nc(CO)[nH]2)C1 c1(CCC(=O)NCC(CCOC)NC(C2(OC(C)C)CCCC2)=O)c(C)n[nH]c1C N1(C(CC(CC)C(F)F)=O)CCC2(CCCN2C(C2SCCCS2)=O)CC1 c1(CC(=O)NC(C)CN(C)C(C2CC2(F)F)=O)cnn2ccccc12 c1(OC(C(N2CC(CSC)OCC2)=O)C)c(C)cccc1Br N1(C(C)=O)CCC(NC(C2(C(=O)OC(C)(C)C)CCCO2)=O)C(COC)C1 c1(C(N(C2CCCN(C(C3CCCN3N=O)=O)C2)C)=O)ccncc1C(F)F C1(CNC(c2cc(C)oc2)=O)CC(O)CN1C(C1CC2(CC2)CO1)=O C(=O)(C1CCCc2sc(=N)[nH]c21)NC(CNC(c1c(F)ccc(CC)c1)=O)CO O=C1CCCc2cccc(NC(C3(F)CN(C(C4CCC4)=O)C3)=O)c21 c1(C(N2CC3CCN(C(c4c(C)cncn4)=O)CC32)=O)cc(C)cc2c1CCC2 CCC(CC)C(C)C(=O)N1CC(C2CN(C(=O)CC3CCCC(C)(C)O3)C2)C1 C(=O)(C(C)S(N)(=O)=O)N(CCCNC(c1ccc(C(C)C)nc1O)=O)C(C)C C(c1cnn(-c2ccccc2)c1)=CC(=O)NCCCCN(C)C(c1ccns1)=O N1(C(Cc2c(C)cccc2)=O)CC2CCC1C2NC(c1ccc(O)c(CO)c1)=O N1(C(C(CC)(C)C#N)=O)CC(NC(=O)Cc2cccc(COC)c2)CC(C)(C)C1 C(=O)(CCCCN1C(=O)CCC1=O)NCC(CC=C)NC(=O)Cc1cnc(C)[nH]1 C1(C(=O)NC(C2(N(C)C)CCCC2)=O)CC(=O)OC1(C)C C1(COC)CN(C(=O)CNS(C)(=O)=O)CCN1C(c1ccc(F)cc1F)=O c1(C(N2CC3(CC(NC(C(C)NC(=O)NC)=O)C3)C2)=O)cccc2[nH]c(C)cc12 C#CCC(C(=O)NC(CC)C(C)(C)O)NC(=O)CC(C)n1ccnc1 N1(C(c2c(C)nc(O)cc2)=O)CCC2CCN(C(=O)CCCCCC(C)C)C2C1 Cc1csc(=NCC(=O)NCC2CCN(C(=O)CCC3CC3CC3CC3)CC2)[nH]1 c1(-n2c(Cc3c(C)nc(C)o3)nc(C3CCCCC3)n2)ccc2c(c1)OCCO2 c1(OC)ccc(C(C)C(=O)NCC2(CNC(=O)CN3CC(=O)NC3=O)CC2)cc1 S(=O)(=O)(C1(c2cn(CCC(N3CCCC3C(F)(F)F)=O)nn2)CC1)N(C)C C1(NC(c2cc(C)oc2C)=O)CN(C(=O)Cn2cc(Cl)cn2)C2(CCCCC2)C1 C1(NC(c2[nH]ccc2C2CC2)=O)CC(NC(C2CCCOCC2)=O)C(O)C1 N1(C(C=C(CSC)C)=O)CCC(CO)(NC(c2ccc(CCCCO)o2)=O)CC1 C1(CC)CCN(C(=O)COCc2ccncc2)C1C(=O)NC(C)Cc1ccncc1 CCC(CNC(=O)CN(C)CCOC)(CC)C(=O)N(C)CC1CCCC1 C1(NC(c2nc(C(F)(F)F)cs2)=O)CC(O)CN1C(=O)CSCCN1CCCC1 N1(C(C2CN(C(=O)C3=CCCS3)CC(F)(F)C2)=O)CC2CCC(C1)C(=O)N2 Cc1cnc(S(C)(=O)=O)nc1N1CCC(C(=O)NCc2ncc(Br)s2)C(O)C1 N1(C(C(C)OCC2CC2)=O)CC(NC(C2(CCF)CCC2)=O)CCC1C C1(NC(CC(C=C)CC)=O)C2CC3CN(C(c4snnc4C)=O)C1C3C2 C1(NC(c2cccc(N(C)C)n2)=O)CN(C(C2CCS(=O)(=O)C2)=O)C(C)(C)C1 c1(OCC(=O)NC2CCCC2NC(C2CC3CCC3C2)=O)ccc(F)nc1 C(CC(=O)NOC(=O)C(C1CCOC1)OC)N(C(C)C)CCC1CCCO1 N1(CC(=O)NC2(CCCNC(C(OC)OC)=O)CCCC2)CCC(C(C)O)CC1 CCC(F)(F)C(=O)NCCC1CN(C(c2conc2C(C)C)=O)CCO1 c1(N2CCOCC(NC(C3(N(C)C)CCCCC3)=O)C2)nc2ncc(Cl)cc2o1 C#Cc1ccc(C(=O)NCC2CC(NC(=O)Cc3ccoc3C)CC2O)cc1C c1(OCC)n[nH]c(=NC(=O)C(CSC)n2ccnc2-c2ccc(S(C)(=O)=O)cc2)s1 c1(CN2CCC(C#N)(NC(C3(C#N)CCC3)=O)C2)cc(F)c(O)c(F)c1 Cc1cc(C)n(Cc2ccccc2C(N2CCC(N(C(=O)CCF)C)C2)=O)n1 c1(CN2CCN(C(C3(O)CCN(S(C)(=O)=O)CC3)=O)CC2)ccc(C#N)cc1O N1(C(c2cc(C)c(C)[nH]2)=O)CC(C(=O)O)C2(C1)CN(C(C1CC(C)CC(C)C1)=O)C2 Cc1cc(Cl)cc(CNC(=O)CN2CCOCC2(C)CO)c1Cl N1(C(=O)Cc2cccc(F)c2)CC2CCN(C(=O)Nc3ccc(Cl)c(Cl)c3)C2C1 N1(C2CN(C3CCC(C)(C#N)CC3)CC2O)CCC2CCCC2CC1 C(C(F)(F)C(=O)N(C1CC2(CNC2)C1)C(c1ccccc1)C#N)OCC(C)C CC1=C(C(=O)N(CCCNC(c2n[nH]c3cccnc23)=O)C2CC2)CCCO1 C1(CNC(C2CCC(OC)CC2)=O)CN(C(=O)C(C)OC)CCC1(F)F c1(OCC=C)ccc(C)c(C(=O)NCC2CCS(=O)(=O)N2)n1 C=CCC(C(=O)N(CCCNC(C1CSCN1C(C1(C)CC1)=O)=O)C)NC(C)=O N1(C(C(CC)OCC)=O)CCCN(C(=O)C=C(C)c2ccccc2)C(C(C)C)C1 c1(C(N(CC(C)(C)NC(=O)OC(C)(C)C)C)=O)cnn(C(F)F)c1 N#Cc1ccc(C(=O)NCC2CCC(NC(c3nscc3Br)=O)C2)c(F)c1 N1(C(C2CN(C(C(C)NC(=O)OC)=O)C(C)(C)C2)=O)CC2CN(C)CC2C1 C1(N(C(CC=CCC)=O)C(C2CC2C#N)=O)CCN(CC=O)C1.OC Cc1ccc(C=CC(=O)NCC2CN(C(=O)C(F)=C(C)C)CC2C(F)(F)F)cc1 C(=O)(CC(C)(c1cccnc1)NC(=O)CNc1ccc(C(C)(C)C)cc1)OC N1(C(C(CCSC)NC(=O)CCC=C(C)C)=O)CCC12CCCC2 c1(CC)c(OC)cccc1C(N1CCC(NC(c2cc(C)c[nH]2)=O)C(F)C1)=O CC1CC(CO)CN1C(=O)CN(C(=O)Cn1cnnc1)C(C)C C=CCC(C(=O)NC1CCC1NC(=O)CCOc1ccccc1C)NC(C)=O N1(C(C(CSC)OC)=O)CCN(C)C2(CC2)C1 CC1CN(C(=O)Cc2ccc(Cl)cc2)CC1C(=O)Cc1cccs1.C(=O)C=CC=O c1(C(=O)NC2CN(C(c3n(C)cnc3)=O)C3C2C3)cccc2c1COCCN2 N1(C(CC(CC)O)=O)CCCCC(C(=O)NC(C2CCCCC2)C)C1 C1(NC(COC(CC)C)=O)CCCCC1CNC(c1ncccc1C(=O)OC)=O C(=O)(CC(C)C(C)(C)C)NC(C1CCN(C(CCCNC(=O)OC)=O)C1)C N1(C(CNC(CCC(C)C)=O)=O)C2CCCC1CC(NC(=O)CCF)C2 N1(C(C2CC(N(C)CC)C2)=O)CCOCC(NC(C2(C(F)(F)F)CCC2)=O)C1 c1(CN2CCC(CC(=O)NC(CCSC)CO)C2)c(F)c(F)cc(F)c1F C1(OC)CCn2cc(C(=O)OCC3CCC(c4ccccc4)CC3)nc2C1 C1(OC)(CO)CCN(C(=O)C(C)CNC(=O)CN(C)C)C1 C1(NC(CC2(C)CCOC2)=O)CCC(NC(=O)C(F)(F)C2CCOCC2)CC1 N1(C(C2(C)CCCCC2)=O)CC(NC(c2cc3c(s2)CCC3)=O)CC12CCOC2 c1(OC)cc(C(=O)NC2C=CC(CNC(c3cnc(C)s3)=O)C2)ccc1C Cc1ncnc(O)c1C(N1CCC(C(C)NC(=O)C#CC(C)(C)O)C1)=O C=C(CNC(=O)CN1CCSCC1)CCNC(c1ccc(CC)o1)=O C(=O)(C1=NN2CCCN=C2N1)NC1C2CCN(C(CCC3N(C)CCC3)=O)C21 C(=O)(CC(C(C)C)OCC)N1CCCC(N(C(c2ccsc2CC)=O)CC)C1 c1(CC)nc(C)cc(=NC(=O)c2cc(-c3ccccc3)cc(N)c2)[nH]1 c1(C(N(C(CNC(COCCOCC)=O)C)C)=O)ccc2[nH]ccc2c1F N1(C(CN(C(C)=O)C)=O)CCN(C(c2cc(N(C)C)n[nH]2)=O)CC1C1CC1 C(=O)(C1CCSc2ccccc21)NC1CC(CCNC(CC(C)CN(C)C)=O)C1 N1(C(C(=O)NCC(F)F)=O)CC2CN(C(C3C4COCC34)=O)CCC12 c1(C(=O)NC2C(CNC(c3ccc(OC)c(F)c3)=O)CC2)cccc2scnc12 C(=O)(C(O)C(C)(C)C)NC1C(C)(CNC(c2ncc(CC)cn2)=O)CCC1 C(=O)(C(C#N)C(=O)Nc1ccc(-c2ccccc2OC(F)F)c(C)c1)OC c1(OC)ccc(CC(N2CCC3CC23C(=O)NC(c2nn(C)cc2O)C)=O)cn1 C#CCC(CC(F)F)C(=O)N(CCCNC(C1NC(=O)OC1(C)C)=O)C N1(C(CC(C=C)C)=O)C(C)CC2CN(C(c3coc(C4CC4)n3)=O)CC12 C(=O)(CCCC(C)=O)N(CC(CNC(C(c1ccc(C(F)F)cc1)OC)=O)C)C n1(CC(=O)NCCOCCNC(C=CC(=O)OC)=O)ccc(-c2ccccc2)n1 c1(C(=O)NC2CCN(C(C3C(CCOC)C3)=O)CC2C)cnc2ncccc2c1 C(C(C(=O)NC1CCCC1C(=O)O)n1cc(C(C)(C)O)nn1)OC(C)(C)C N1(C(CC(C)c2cnn(C)c2)=O)CCC2CC1CN2C(=O)CC(F)(F)F c1(C(=O)NCC2N(C(CC3(OCC)CCCC3)=O)CC2)ccc2c(c1)N(C)CC2 C12CNC(=O)CN1C2=O.C1(CC(=O)NC2C=CCC(CC)C2)COCC1(C)C C1(CNC(C=CC)=O)CCN(C(=O)CNC(=O)CCCCC)C(C)C1 C1(CN(C)C)CCN(C(=O)C(=O)NC(=O)C2CC2)CC1.C12CN(C1)C2 Cc1[nH]nc(C(N2CCCC(N(C(=O)CCNC(C3CCC3)=O)C)C2)=O)c1O C1(N(C(CC(CC)C2CC2)=O)C)CCCN(C(c2cnccn2)=O)CC1 C1(NC(CC(c2ccc(CC)cc2)C)=O)CC2CN(C(=O)C=CC3CCC3)CC12 C1(C(=O)NCCC2(O)CN(C(=O)C(c3cncnc3)C)C2)(SC)CC(O)C1 c1(C(=O)NCCN(CCC)C(C2CCC(C(=O)OC)C2)=O)csc(Cl)c1OC Cc1ccc2ncc(C(=O)NCC3(F)CCC(NC(=O)C(C)C(C)(C)C)C3)n2c1 N1(CC(N)=O)CC(NC(=O)CCCC2CCC2)CC2(CCOCC2)C1 C1(NC(c2cnc(OC)c(Cl)c2)=O)CCCC12CCN(S(=O)(=O)C(F)(F)F)C2 C1(CC)(CC)CC(NC(c2ccnc(C)c2)=O)CN1C(c1ccoc1)=O C(CC(C)(C)C(=O)N(CCNC(C1CCOC1C)=O)C(C)C)SC C(=O)(CCC(=O)c1cccs1)NCc1scnc1C.c1(C)nn[nH]c1C(=O)N(OC)CC C#CC(CNC(=O)CC1CC(NC(=O)COCCO)C1)COCC.OCC n1(CC(=O)NC(C2CC(NC(C(CCCC)O)=O)C2)C)ncc2ncccc12 C1(C)(C(N(C2CCN(C(CC(C)C)=O)C2)CCO)=O)CC2CCC(C1)S2 C1(O)(CNC(CC(C)(C)SC)=O)CCCN(C(C2CCCN(C)C2)=O)CC1 c1(C(N2CCC(F)(C(=O)NCCc3ccncn3)C2)=O)ccc(F)cc1Br C#CCC(C)(C(=O)N1CCCCCC1CCO)NC(=O)CCc1cnco1 CCCCCCCCCCCCCC(=O)NCC1(C)CCN(C(C2CC2C)=O)C1 CCC(CCC(=O)NC(c1nccc(C)n1)C)NC(c1cc[nH]c(=NC)c1)=O C1(CC)CN(C(c2coc(N(C)C)n2)=O)CCC1NC(=O)CCNC(C)=O C12(CNC(c3ccccc3OCC(F)(F)F)C(F)(F)F)CCC(CC1O)C2 C(=O)(C1=C(C)CC(C)(C)CC1)N1CC2C(NC(c3cc(CCC)n[nH]3)=O)(CC2)C1 c1(C(=O)NC(c2ccccn2)(CC)C)cc(COC)on1 c1(C(=O)NCCC2CCN(C(C(C)OCC(C)C)=O)C2)ccc2cc[nH]c2c1 N1(C(C(=O)Nc2c(CC)oc(C)c2)=O)CCCc2c(Br)ccc(OCC)c21 C(=O)(CCCC(=O)NC(C)C)NCC(CNC(c1cncc(C)c1)=O)O N1(C(C)=O)CCc2ccccc2C1CC(=O)NCc1cnc(C(F)(F)F)s1 N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(=O)CCCn3cccn3)CC12 S(=O)(=O)(c1ccccc1[N+](=O)[O-])NC(c1cccc(Cl)c1)C(N1CCOCC1)=O c1(CN2C(C(C)O)CCCC2)ccc2[nH]nc(Cl)c2c1 CCC(C(C)(C)O)NC(C1CN(C(c2ccnc(C)c2)=O)CC1C)=O c1(CC(=O)NCC2CC(NC(C(c3ccn(C)n3)C)=O)C2)cccc(Br)c1 C(C(C)C(=O)NCC=CC1CCCC1)(C1CC1)NC(=O)OC(C)(C)C N1(C(Cc2ccc(C)cc2)=O)CC(C2CN(C(c3cncnc3C3CC3)=O)C2)C1 C1(C(=O)NCCC#N)CC2(CCN(C(c3[nH]cc4c3CCC4)=O)CC2)CO1 c1(OC)ccc(-c2ccccc2CN2CCN(c3ccncc3)CC2)cc1O Cc1ccc(Cl)cc1OCC(=O)NCC1CCCN1C(=O)C#CC1(C)CC1 C(C)(C(=O)NC1(NC(=O)C2=CCCOC2)CC1)(C(C)C)Nc1ccc(C)cc1 C(=O)(C1=CCS(=O)(=O)C1)NCC1CCCCN(C(c2cc(C)c(C)[nH]2)=O)C1 C(C(=O)N=c1cc2ccccn2[nH]1)(C1CCCC1)NC(C(C)(C1CC1)NC(C)=O)=O C12(NC(CSC)=O)CC(CSC3CN(C(=O)COC(F)F)C3)(C1)C2 N1(C(C2CCCC(C#N)C2)=O)CC2(CCN(C(=O)CCn3cnnn3)CC2)C1 C1(C)(NC(C2CC(C)(C)C2)=O)CCN(C(=O)C(F)(Cl)c2ccccc2)C1 CC1CN(C(c2cnn(C)c2Br)=O)CCCN1C(c1cc(C#N)n(C)n1)=O C1(C(=O)NCCCCN(CC)CC)CN(C(=O)C(CC)SC)CC12CC2 c1(C(N(CC(C)(C)CNC(C2(OC)CCCOC2)=O)CC)=O)cc(F)ccc1F C1(CC)CN(C(C2(c3ccccc3Cl)CC2)=O)CCN1C(c1ccn(C)n1)=O c1(C(C2CCCC2)NC(CSCC(COC)O)=O)ccccc1F N1(C(C2CCC(=C)CC2)=O)CCC2CCCN(C(=O)CC3CCC3)C2C1 N12CCC(CC1)C2.c1(NC2(C3N(C(C(C)OC)=O)CCC3)CC2)cc(C)ncn1 FC1(F)CCC(n2nc(-c3ccsc3)nc2CCc2cc[nH]n2)CC1 CC1C(=O)N(CC(=O)NC2CN(C(c3cnn(C)c3)=O)CC2(C)C)C(=O)C1C C(=O)(C(O)C(C)(C)C)NC(C)CC1CN(C(C2(CC3CCC3)CC2)=O)C1 c1(C(=O)Nc2cc(C)c(NC(C34CC5CC3C4C5)=O)cc2)cccc2ncn(C)c12 N1(C(c2ncc(OC)cn2)=O)CCCC2(C1)CN(C(=O)C(c1ccc(C)s1)C)C2 C=CCC(CNC(c1ccc(C)s1)=O)NC(c1cc(C(F)F)[nH]n1)=O Cc1cc2c(cc1C)C(C(=O)N1CC(NC(C3(C)CC3(F)Cl)=O)C(C)C1)CO2 C=CCC(C)(CC=C)NC(C1(CNC(=O)C(C)CO)CC12CCC2)=O C1(C(=O)NCC2CCCCC2NC(C2(O)CC2)=O)CC2(C1)CC1(CC1)C2 CS(=O)(=O)CCC(=O)NCCC(O)C(=O)N1CCC(N2CCC2)C1 CCC(C)(CNC(c1cc(C)nnc1C)=O)C(=O)N1CCCC(CCO)C1 c1(CNC(c2ncc(CC)s2)c2nnnn2CC)c(F)cccc1Br Cc1ccc(Cl)cc1Cc1nc(-c2cccnc2)nn1-c1cccc(Cl)c1 N1(C(c2nc(CC(C)C)sc2)C(=O)NCCC#N)CC(C)C12CCOCC2 c1(CC(=O)NC2(CN(C(=O)CC3CCOC3)C)CC2)ccnc(Br)c1 C1(C(=O)NC2CCN(C(C3CCS(=O)(=O)N3)=O)C23CCC3)CC2(C1)CS(=O)(=O)C2 CC(C)CC(F)C(=O)N1CC(CNC(=O)CCCCCc2cccs2)CC1C N1(C(c2c(CC)nns2)=O)CC(C2CCCN(C(c3nccc(CC)c3)=O)C2)C1 c1(SCC)cccc(N(C(=O)C(C2CCOCC2)OC=O)C)c1.C1(O)CCCOC1 c1(OC)cc(N)ccc1C(N1CC(O)(C(C)NC(C2CNC(=O)N2C)=O)C1)=O C1(CNC(Cc2nc(C)sc2C)=O)CN(C(=O)CCc2cccn2C)CCCO1 C#Cc1ccc(Cl)c(C(N2CCC3(CC2)CC3NC(=O)COC)=O)c1 N(C(=NCC1CC1)N1CCS(=O)(=O)CC1)C(C)Cc1ccccc1 C(=O)(CC(CC(C)C)COC1CCCC1)NCC(CO)O.C(=O)(CO)CC c1(CSC)cccc(C(N2CCC(F)(CNC(c3c[nH]nc3C)=O)C2)=O)c1 C1(CNC(C(CCC)OC)=O)CN(C(=O)CCc2ccc(F)cc2)CC(C)(C)O1 C1(CNC(C(C)n2ccnc2)=O)CC2CCCC2N1C(C1CC(O)C1)=O c1(OC)cccc(SCC(N2CC(CNC(=O)C(F)=C(C)C3CC3)CC2C)=O)c1 N1(C(=O)NC(n2ccnc2C)CC)CC(C#N)CC1CC C(=O)(CCCCC1CC1)N1C(C2(C)CC2)CCC1.c1(C(=O)N)cn(C2CC2)cn1 C1(CNC(C2C(C)OC(C)C2C)=O)CC(N=c2[nH]c3ccc(O)cc3s2)C1 N1(C(C(C(C)C)CNC(=O)COCC2CCOC2)=O)CC2(C)CCC2(C)C1 C1(CN(C(=O)CCNS(C)(=O)=O)C)CCCN1C(c1nc(Cl)cs1)=O c1(C(=O)NCCCN(C(c2cc(Cl)nnc2Cl)=O)CC)nc(C)n2ccccc12 c1(CC(=O)N(C2CCCN(C(=O)C(O)CC(N)=O)CC2)CC)ccc(C)c(C)c1 c1(C(=O)NC(C#C)CC(C)C)cc(Br)cc2nc[nH]c12 C1(NC(c2cnc(C(C)C)[nH]2)=O)C(C)CN(C(=O)CC2(CN(C)C)CC2)CC1C CC(C)CC(=O)C(=O)NCCn1cc(C(=O)NCC2CCCC(F)C2)cn1 N1(C(CCc2c(C)noc2C)=O)CC2CC1CN(C(C1(C)CCCN1C)=O)C2 Cc1ccc(-n2nc(-c3ccncc3)nc2CCN2CCOCC2)cc1C C1(N(C(=O)CC2CC2(C)C)C)CCC(NC(=O)CC2CCCCC2)C1 c1(OC(C)C(=O)NC(C)CN(C)C(c2cc(Br)co2)=O)ccc(F)cc1 CCC(CC(=O)N1CC2CC1C2CNC(C1CC1c1cnn(C)c1)=O)C(C)C S(=O)(=O)(c1c[nH]ccc1=NCCc1ccc(Cl)cc1)NC1(CC)CCCC1 C1(C(=O)NC2(CNC(C(C)OCC3CC3)=O)CCCCC2)CCC(C)(F)CC1 C1(C2CCCN(C(=O)C(c3ccccc3Cl)O)C2)(NC(C(C(C)C)O)=O)CC1 c1(C(CC(=O)NCC2(OC)CN(C(C3CCCC3(F)F)=O)C2)C)c(C)noc1C c1(CN(C=O)CC2(NC(N)=O)CCOC2)cc(C(F)(F)F)cc([N+](=O)[O-])c1 N1(C(c2cc(SC)oc2C)=O)CCN(C(=O)Cc2ccc(Cl)cc2)C2CCCC12 N1(C(C2CC(=O)N(CC(C)C)C2)=O)CC(NC(C2C(COC)C2)=O)C(C)C1 CC(C)(CCC#N)C(=O)N1CCCCC(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(=O)NC2C(CNC(C(Cc3c(C)nc[nH]3)O)=O)C2)ccc(C(O)CF)cc1 C12(CNC(Cn3ncc(CC)c3)=O)CCC(C1)N(C(C1CCCC1O)=O)C2 C12(NC(CC(CC)OC)=O)CCOCC1CN(C(c1cnco1)=O)C2 C(=O)(CC(=O)NC(N(CC(C1CC1)OC)C)=O)N.C1(C(C)NC2CC2)(CS)CC1 C(=O)(CCC1=NNC(=O)CC1)NCCN(CCC)C(C1(F)CCCOC1)=O c12ccc(s1)C2.N1(C(C)=O)CC=CC1CSC(C(=O)NC(c1ccco1)=O)C C1(NC(C2(C(F)F)CCN(C)CC2)=O)Cc2n[nH]cc2C(C(F)(F)F)C1 N1(C(COCC)=O)CC2COCCC2(NC(=O)CC(=O)NCc2ccccc2)C1 N1(C(c2ccc(CCC=C)cc2)=O)CCCCC(N(C(=O)C(N)=S)C)C1 CCC(C)C(C)C(=O)N1CCN(C(=O)OC(C)(C)C)CC1Cc1ccnc(Cl)n1 C1(CNC(CNC(=O)OC)=O)CCC(C)CN1C(C1CC2C=CC1O2)=O C1(C(=O)NCCn2cnc(C)c2C)CCN(C(c2cnc(C(C)C)o2)=O)C12CC2 CC1(C)CC(NC(c2ccc(-n3cnnn3)cn2)=O)CN1C(C1CC2(CC2)C1)=O C=CCCC(C(=O)NCc1cc(C)c(C)o1)NC(c1cnncc1O)=O C(CCCC(=O)N1CCCCC1CN(C)C(c1occc1F)=O)SC CCC(C)CCC(O)CC(=O)N1CCN(c2nccc(C#N)n2)CC1 c1(C(=O)NCC2C(C)CCN2C(=O)C(=O)NCC2CC2)c(F)cc(Cl)cc1Cl C1(NC(c2c(C)cc(CO)o2)=O)CN(C(c2ccc[nH]2)=O)CC1N=[N+]=[N-] c1(C(=O)NC2C(C)CN(C(c3ncc(Br)cn3)=O)C2)cc2c(ncn2C)[nH]1 C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(C1CC1)NC(Cc1noc(C)c1C#N)=O C(C(=O)NC(CN(C)C)C(C)C)(C(C)C)NC(c1nc(CCC)oc1)=O N1(C(c2n(C)cnc2)=O)CC(C2CCCCN(C(=O)NC3(C)CC4CC4C3)C2)C1 C12(C(N(C3CCC(NC(c4n(CC)ncn4)=O)CC3)C)=O)CCOC1CCOC2 c1(C(=O)NOC2CCOC2)ccn[nH]1.c1(C)ccccc1 C(N=c1cc(C)nc(N2CCC(NC(C)=O)C2)[nH]1)c1c(OCCC)cccc1 O=C(O)CCCCC(=O)Nc1ccnc(OC2CCOC2)c1 c1(CCC(=O)NC2C(NC(C(=C(C)C3CC3)F)=O)C2)ccc(O)cc1 C(CCCCC(=O)NC1CCOC1C1CC1)n1cc(COCC(=O)OC)nn1 CN1CCOC2(CN(C(c3n[nH]cc3CNC(C3CC=CCO3)=O)=O)C2)C1 O=C(C1=NOC(CNC(C23C=CC(CC2)C3)=O)C1)Nc1ccc(Cl)c(O)c1 Cc1cnc(CC(=O)NCC2(C)CCC(NC(c3ccc(CO)o3)=O)C2)cn1 c1(N(C)CCn2cnnc2)nnc(N2C(=O)CC(Cc3cnccn3)C2)n1CC N1(C(c2cnc(C)s2)=O)CCN(C(=O)COc2cccc(CO)c2)CC2(CC2)C1 C1(NC(COC(CC)(C)C)=O)CC2CC1CN(C(C1(CO)CCCO1)=O)C2 C1(CNC(c2nc(C)n(C)n2)c2nnnn2C)CC2CCC(C1)C2 Cc1ccccc1NCC(=O)NC1(C)CCN(CCCC(C)(F)F)C1 CN1CCOC(C(=O)NCC2CC3CCC2N3C(C2(C(N)=O)CCC2)=O)C1=O N#Cc1cc(C(N2CCC(O)(CNC(c3cc(F)n[nH]3)=O)C2)=O)cc(O)c1 N1(C(CC(C=C)C)=O)CCCC(C)(C(N2CC(C3(C)CC3)C2)=O)C1 C(=O)(C1CCc2nccn21)NC1(COC)CN(C(=O)CC(C)CC(C)(C)C)C1 N1(C(C2CC3(CN(C(c4cccnc4S)=O)C3)OC2)=O)CCc2ncncc2C1 C1(NC(C(CC)O)=O)(CNC(=O)C(c2ccc(C)cn2)(F)F)CC2CCC1CC2 C1(C(N(CCCC)C)=O)CNC(=O)CN1C(C1CC1CC(C)C)=O c1(CC(=O)NCC(CO)NC(c2c(CCC)onc2C)=O)c(C)nc(C)nc1O c1(CC(N2CCCCC2Cc2cn(C3CCOC3)nn2)=O)ccc(F)c(Br)c1 N1(C(c2c(NC)cncc2)=O)CC=C(C(=O)NCC2CCC(C)(C)CO2)C1 c1(OC)c(C(=O)NCC2CN(Cc3cnc(C)s3)CCO2)cccc1C(F)(F)F n1(CC)c(C(=O)NCC=CC(=O)N(C(C)CCc2cn[nH]c2)C2CC2)cnc1O c1(C(N2C3CN(C(C(C)(C)Br)=O)CC2C3)=O)ccc2c(c1)CCC2 C1(NC(CC(C)F)=O)CCCC(C(=O)NCC2(O)CCC2)C1 C1(CC)CC2(CCN2C(C2CCN2C(C2(OC(C)C)CCC2)=O)=O)C1 C12(NC(c3cnccc3Cl)=O)CCN(C(=O)COCC(F)F)CC1C2 N1(C(C(=O)NC(CC)(C)C)CCOCCO)CCNC(=O)C1(C)C c1(C(=O)NCC(CNC(c2nn(C)cc2Cl)=O)OC)ccnc(Cl)c1N Cc1nnn(CC(=O)NC2C=CC(CC(=O)NCCc3nccs3)C2)n1 c1(C(=O)NC(CNC(C(C)N(C(C)=O)C)=O)CO)ccnn1C(C)C c1(SC)cc(C(=O)NCCCCC(C)NC(=O)Cc2ccnn2CC)ccc1F CC(CCCO)NC(=O)CC1CC(NC(=O)CCn2cnnn2)C1 c1(C(C)NC(C2CC(CCC)C2)=O)nocc1C(=O)NCC(C)(C)CO C1(NC(C(F)=C(C)C)=O)CCN(C(c2cnn(-c3ccccn3)c2C)=O)CC1C CC(CC(=O)N1CCC1CNC(=O)Cc1ccc2occc2c1)C(F)(F)F c1(C(=O)NC(C)CNC(c2cc(C3CC3)ns2)=O)cccc(S(N)(=O)=O)c1 CC(C)C(C#N)C(=O)NC1(CCCNC(=O)CC2CCC(=O)N2)CC1 C1(CNC(C=CCCC)=O)CC(C)N(C(c2cccc(OC)n2)=O)C1 c1(C(N(C2CCCC2)CC)=O)c(CNC(=O)Cn2nccn2)cnn1C c1(CC)nnc(C(=O)NCC2CCCN2C(=O)C(c2ccccc2)N(C)CC)s1 N12CC3CN(CC3C1)C2=O.c1(C(N2CCC(c3ccccc3)C2)C)ccccc1S CCC(CC(=O)NC1CCCCC1NC(C1(C)CC(F)(F)C1)=O)SC N1(C(c2cn(CCCC)nn2)=O)CC2(CCC(CNC(=O)CC(F)(F)F)O2)C1 c1(C(N2CC(C)(OC(CCC)C(=O)NCC)C2)=O)ccc2nnc(S)n2c1 CN1CC2CCCC(C1)N2C(C1(C)CCCN1C(C1CCOCCC1)=O)=O c1(C(=O)NCCCCNC(C(c2cn(C)nc2)O)=O)ccc2c(c1)OCC2 C1(CCC)(C(=O)NCCCCC(C)NC(c2cc(C)sc2C)=O)CCNC1=O C1(C(N2CCC(OC)C(F)C2)=O)C(C2CC2)CCN1C(c1ccsn1)=O C1(NC(c2c(OC)ccs2)=O)CCCC(NC(c2ccc(C3CCC3)cc2)=O)C1 N1(C(C2N(C)CCC2)=O)CCN(C(C2(N3CCCCC3)CC2)=O)CC1CO c1(NCCCC)ccc(S(=O)(=O)N2CCC(C)C(CO)C2)c(Cl)c1 N1(C(CCC=C)=O)CCC2CCCC(C1)N2C(=O)C(C)Oc1ccc(Cl)c(Cl)c1 CC(C)(C)C(=O)N1CCCC1C(N1CCC1CNC(c1ncc(C(N)=O)o1)=O)=O c1(CC)nc(=N)[nH]cc1C(=O)NC(C)CC(C)NC(c1cc(Cl)c(Cl)n1C)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)CCNC(=O)Cn1ncc2cccnc12)C N1(C(c2ccc(SC)s2)=O)CC(NC(c2ccc(N)c(F)n2)=O)C(C)(C)C1 c1(CN(CC(C)O)Cc2c(C(=O)OC)ocn2)ccc(F)cc1F C(=O)(CCCC(=O)NCCCOCCNC(C1CCCC(C)C1)=O)NCC N1(C(C2CCCOC2)=O)CCN(C(c2cc(Cl)cc(Cl)c2)=O)C(CO)C1 C1(C(CC)NC(C2(C)CCOC2)=O)CCN(C(=O)C=Cc2ccccc2)CC1 C1(NC(C(CC(=C)Cl)NC(=O)C(C)COC)=O)CN(C)CCN(C)C1 C=CCC(C(=O)OC)c1ccccc1.C1(CCC)CN(C(c2nnnn2CC)C)C1 N1(C(C(C)n2ccnn2)=O)CCC(N(C)C(c2csc(Cl)c2)=O)C2(CC2)C1 Nc1ccc(Cl)cc1C(N1CCCN(C(C23CCCC2(C(=O)OC)C3)=O)CC1)=O n1(CC)ccnc1-c1ccccc1.N12CC(C1)C(=O)N(CC)C(=O)C2.C(=O)(CSC)O c1(C(N2CCN(C(C=CC)=O)C(CCC)C2)=O)c([N+](=O)[O-])cnn1CC(F)F N1(C(C(=Cc2cccnc2)C)=O)CCN(C(C2CCCOC2)=O)C(CCO)C1 N1(C(C(n2c(C)ncc2)C)=O)CCC(C)(C)C(C(=O)Nc2cnccc2Cl)C1 Cc1cc(=NC(=O)C(=O)N2CCOCC2CN(C(=O)CC(C)CC(C)C)C)[nH]o1 N#Cc1cccc(C(=O)CN(CCCCN2CCC(O)C2)C)n1 O=C(CCCCCn1cc(-c2cnsc2)nn1)N1CC2CC2C1 N1(C(CC=CCC)=O)CCN(C(c2c(Cl)sc(C)c2C)=O)CC1C1CCC1 c1(OC)ccc([N+](=O)[O-])cc1C(N1CC2CC2(NC(=O)COC(F)(F)F)C1)=O CC1(C)CC(C(N2CCC(NC(c3cc(Cl)cs3)=O)C(O)C2)=O)C(C)(C)O1 C12(C(=O)NCc3ncc(CNC(c4cc(CCO)on4)=O)s3)CCC(CO1)C2 N1(C(c2n(CCC)ccc2)=O)CCOC(CCCNC(=O)Cc2cccs2)C1 Cc1cc(C(=O)NC(C)CCCNC(c2[nH]nnc2C)=O)c2ncccc2c1 C(=O)(C(O)CC(C)(C)C)NC1CCC(N(C)C(c2ccc(C(F)F)cn2)=O)CC1 N1(SC(C)=O)CC2CCC(C1)C2CC(N1CCC(F)(F)CC1)=O.C CCC(CC)CCCC(=O)N1CC2(CC2)CC1CNC(c1nc(C)nn1C)=O N1(C(CC(C(C)OC)NC(=O)CC2CC2)=O)Cc2ccc(C)nc2C1 Cc1ncc(C(=O)NC2CC(C)N(C(=O)CC3CCCCN3C)C2)c(C(C)C)n1 c1(OC)ccc(C(=O)NC2CC2NC(=O)CCN2CCC2)c(C)c1OC N1(C(CC(=O)OC)=O)CC23CCCC2(C1)CN(C(=O)C(C)c1ccsc1)C3 c1(OC)ccc(-c2nc(C)c(NC(N3CC(F)CC3C#N)=O)s2)c(C)c1 N12CCc3nn(C)c(c3C1)C2=O.c1(NC(C)=O)cccc(CNC2CC2(F)F)c1 N1(C(c2scc(OC)c2)=O)CCS(=O)(=O)C(CCNC(C2CCS(=O)(=O)C2)=O)C1 C1(C(=O)NC2(CCO)CN(C(CCC3C(C)(C)C3)=O)C2)CC2(CCC2=O)C1 C1(C(C(=O)N(C(C)CSC)CC)C)CCCN(C(c2cnn(C(C)C)n2)=O)C1 CP(C)(=O)C1CCCCC1C(=O)NC1CN(C(C2(C3CC3)CC2)=O)C1 C1(NC(c2ccncc2Cl)c2n(C(C)C)nnn2)CCCCCCCCC1 N1(C(C)(C)C)CC(CNC(=O)CC2(C)CN(C(=O)CC(=O)OC(C)(C)C)C2)CC1=O C1(CC(=O)NOCCCO)CCCN(C(c2ncccc2Cl)=O)C1 C1(NC(C(CC)OC)=O)CN(C(c2ccc3nc[nH]c3c2)=O)C2(CCCC2)C1 c1(C(=O)NC2C(NC(Cc3ccc(CCC)cc3)=O)C2)cc(F)c(F)cc1F c1(NC(=O)NC2(c3nc(C)on3)CCC2)c2c(nn1C)CCCC2 c1(NC(C)=O)c(F)ccc(-c2cccc(NC(C3CC(O)CN3)=O)n2)c1F C1(NC(C23CC(NC(Cc4nc(C)oc4)=O)(C2)C3)=O)CCOCC1C c1(C(=O)OC)ccccc1C(=O)NC(C)C(C)NC(C1CCC(C(C)C)CC1)=O c1(CC)ccnc(C(=O)NC2(C(=O)OC)CCOC2)c1 C1(CCNC(c2ccncn2)=O)CCN(C(C2CC2c2ccco2)=O)C1 C1(CNC(C(CC)F)=O)CN(C(c2ncnn2C2CCOCC2)=O)CC(C)(C)O1 C(=O)(CC(O)CC(C)(C)C)N1CC(OC)C(NC(c2nnc3ccccn23)=O)C1 CC1CCC(CNC(=O)C(c2ccco2)NC(C2CCC2)=O)N1C Cn1cc(C2OCCC2C(=O)NCCN(C(=O)Cc2ocnc2CO)C2CC2)cn1 CCCC(C(=O)N1CC(CC(=O)NC(c2ccccc2O)C)(OC)C1)N(C)C C(=O)(C1=CCC2CCC1N2C(C1(C#N)CC1(C)C)=O)N(CCF)CC c1(C(N(CCC(=O)NC2CCCOC2)CC#C)=O)cccnc1C N1(C(=O)NC(C(=O)OCC)C2CCC2)CCCC1CNC(=O)CSc1nc[nH]n1 CCCC(N=c1[nH]c(=NCCC2(CO)CC2)c2sccc2[nH]1)c1ccco1 C1(NC(C2(CC#C)CCCC2)=O)CCN(C(C2(CCCC)CC2)=O)CCC1CO C(=O)(C1=CC2CCCCCCC12)N1CC(C)C(CNC(=O)C=CCO)CC1 c1(C(N2CC(O)(C(C)NC(=O)CC(C)(O)C3CC3)C2)=O)cccc([N+](=O)[O-])c1 N1(C(Cc2n(C)ccn2)=O)CC2CC1CN2C(=O)CC1CCOC(C)(C)C1 C#Cc1ccc(Cl)c(C(=O)NCCC2(NC(C3CN(C)C(=O)N3)=O)CCCC2)c1 CCC(C)CCC(=O)NCC1CN(C(=O)Cc2cnc[nH]2)CC1C(F)(F)F c1(CC(=O)NC2C(NC(CCC=CC(C)C)=O)COC2)c[nH]c2ccc(F)cc12 C1(CC=C)CCCN(C(C2CC3CC3N2C(c2[nH]cnc2C)=O)=O)C1 c1(N2C3CN(C(C4CCCN(C)C4)=O)C(C3)C2)nc2cccc(Cl)c2s1 c1(C(N(C)CC2CN(C(c3cnc(SC)nc3O)=O)C2)=O)cc2n(n1)CCCO2 c1(C(=O)NC2(C)CCCN(C(C3CCC4CC34)=O)C2)cn2cccnc2n1 C1(C(N2CC(F)(CNC(C3=C(C)CCCC3)=O)C2)=O)CC(C)c2nc(C)cn2C1 c1(NC(=O)OC(C)(C)C)ccccc1C(C)NCc1n(CC(C)C)ncc1 Cc1nc2cc(C(=O)NC3CC3NC(=O)C(c3cncn3C)O)c(F)cc2[nH]1 CN1Cc2ccc(CNCc3noc(-c4ccc(Br)cc4)n3)cc2C1=O Cc1nc(-c2c(C)noc2C)sc1C(N1CC(CC(C)NC(=O)C(O)C2CC2)C1)=O C1(OCC(=O)NCCC(C)N(C(C(C=CCCC)O)=O)C)CCC(F)(F)CC1 C=CCCCC(=O)N1CC(O)(C(C)(C)CNC(c2c(C(C)C)cnn2C)=O)C1 c1(NC2(CNC(c3cnc(C(C)O)s3)=O)CC2)ncc(Br)c(O)n1 C1(CCNC(C2ON=C(C)C2)=O)CCCN(C(c2ccc(CO)s2)=O)C1 C(=O)(C1=CC2(CCOCC2)C1)NCCC1CCCN(C(C(CC)CO)=O)C1 N1(C(c2ncccc2Cl)=O)CCC2CC2(C(=O)NC2CCN(CCF)C2)CC1 c1(C(N2CCC3(C(NC(CCC(=O)NC)=O)C3)CC2)=O)cc(C)cc2c[nH]nc12 c1(OC)ccnc(C(=O)NC2CC(CCNC(c3cscc3SC)=O)C2)c1F Cc1cc(C(C)C(=O)NC2COCC2NC(=O)CNC(c2cccs2)=O)c(C)o1 C1(SCC(=O)NC2CCN(C(C3(C4CCCCO4)CCC3)=O)C2)CCOC1=O c1(OCC=C(C)C)ccccc1CC(=O)NCC(C)N(C(=O)Cn1ccnn1)C CC1CC2(CCN(C(=O)C3=CCSC3)CC2)CN1C(=O)C=Cc1cccnc1 C1(C(=O)O)CCC2(CCN(CC3CC4(C3)CC(CF)C4)C2)C1 Cc1ncc(CC(=O)N(CCCNC(C2C=CCC2)=O)C(C)C)[nH]1 c1(C(N(C)CCOCCNC(=O)CC2CCC=CCC2)=O)cc(N)ccc1Cl C(N=c1ccc(S(=O)(=O)N(C)CCc2ccc(F)cc2)c[nH]1)c1cc(CC)on1 CC1CN(C(=O)C(O)CNC(C2CN(C3COC3)C2)=O)CC1(C)CO c1(C(N(C)CC2N(C(C3C(C)SCCC3)=O)CCC2)=O)ccc2c(c1)NC(=O)C2 C1(O)(CNC(CC(C)SC)=O)CC2CCC1O2.c12occc1C(=O)NC2 C(C(C(=O)NCc1nccnc1C)C(C)C)NC(C(CC=C)C)=O N1(C(=O)Cc2ccsn2)CCC(C2CC(NC(=O)C(F)(F)C3CCOCC3)C2)C1 CON(CCC(=O)N1CCC(C)(C)C1C)C(=O)Cn1cccc1 Cc1cccc(SCC(N2CCCC2CN(C)C(c2coc(C#N)c2)=O)=O)c1 c1(CC)onc(C2CCCC2)c1C(=O)NC(C)CC(C)NC(C1CCCS1)=O N1(C(c2cncc(COC)c2)=O)CC2CCC1CN(C(c1ccn(C)c1C)=O)C2 N1(CC2(C)CC3(CCC3)C2)CCC(=O)N(CC2CCCO2)C1=O Cc1nnccc1C(=O)NC(C)CC1CCN(C(C2(Cl)CC2)=O)CC1 C1(N(C(C=CC(=O)NC)=O)C)(CC)CCCN(C(=O)CC(C)N(C)C)C1 C1(CC(N2C(C)(CC(=O)NCCc3c(C)ncs3)CC2)=O)CCC(C)(C)C1 N1(C(C2CCC(C)O2)=O)CCCN(C(c2occc2F)=O)C(C)C1 C1(C(=O)NC(CC)C(N)=O)CCN(C(c2ccc(O)nc2C)=O)C(C)(C)C1 C1(C2CN(C(c3cccc(F)c3SC)=O)C2)(NC(C(CSC)OC)=O)CC1 c1(C(=O)NC2CN(C(C34CCC(CC3)CC4)=O)CC2(F)F)ccc(F)cc1Br N1(C(C2CCC(NC(C)=O)CC2)=O)CC2(CC2)CC1CNC(C1CCC(C)O1)=O CC(CC(=O)N1CC2(CCCN(C(c3ncncc3Cl)=O)C2)C1)CC(C)(C)C c1(OC)nc(C)ccc1CNC(c1ccc(C(N2CCCC(C)C2)=O)cc1)=O C(CC(CC)C(=O)NC(C)CN(C)C(c1cc(C2CCOCC2)no1)=O)=CC N1(C(c2cc(=NC)[nH]cc2)=O)CCN(C(C2CCC(O)C2)=O)CC(O)C1 c1(-c2nc(C)sc2)cnc(N)c(O)c1.c1(C2CC2)ccc(Cl)cc1C C1(N(C)C)CC(NC(=O)CCCNC(=O)C=Cc2ccncn2)C1(C)C C(N=c1ncnc2[nH][nH]c(Br)c1-2)N1CC(N2CCN(C(C(C(C)C)=O)=O)CC2)C1 C(C(=O)N(CCC(C)NC(c1ccccc1F)=O)C)(C(C)C)SC c1(C(N2CCC(NC(c3ccc(OC)o3)=O)C2)=O)nccc(Br)c1C c1(NCCC(C)N(Cc2ccc(F)cc2F)CN)ccc2c(c1)CN(C)C2.N(C)C C1(C(N2CCC(C(N)=O)C2)=O)COCCN1C(C1CCCCO1)=O C#CCCCC(C)C(=O)NC1(C(=O)Nc2ccnnc2O)C(OC(C)(C)C)CC1 c1(C(N2CCC(CC=C)(NC(=O)CCC(=O)OC)C2)=O)cccn2cncc12 n1(CCCC)nnc(C)c1S(=O)(=O)N1CC2(C1)CC(C)(C)C2 Cc1cn2nc(C(=O)NC3CC(C)(NC(C4CCCC(F)C4)=O)C3)cc(C)c2n1 C1(NC(c2c(OCC)scc2)=O)CCCC12CN(C(=O)COC(C)C)C2 C1(CNC(C=CC)=O)CCN(C(=O)Cc2cc(Cl)cc(Cl)c2)CC1O N1(C(=O)OC(C)(C)C)CC2CCC(N=c3ccn(-c4ccc(F)cn4)[nH]3)C2C1 C12(NC(C3Cc4cccnc4C3)=O)CC3CCC(C1C2)N3C(C1(F)CCC1)=O n1(C(C)C(=O)NCCCCNC(c2cc[nH]n2)=O)cnc(C#N)n1 C12(NC(CCCC(=C)C)=O)CCCN(C(=O)C=Cc3ccccc3F)CC1C2 C(=O)(C(CC)C(F)(F)F)NCc1n(CC)ncc1.C1(C(=O)OCC)(OC)CCOCC1 C(C(C)(C(=O)Nc1cccc(F)c1)NC(=O)CCCSc1ccccn1)SC Cc1cc(C)c(S(=O)(=O)Nc2cnnn2C2CC2)cc1-c1cccs1 C#Cc1ccc(C(N2CCN(C(C)(C)C)CC2)=O)cc1.N12CC(C1)C2=O C1(CNC(=O)CO)C2CN(C(c3cc(Br)n[nH]3)=O)CC12 Cc1ccc(OC(C2CC2CC(C)C)=O)c(F)c1 O=C(C1=CCOCC1)NC1C2CC3C1C3C2C(=O)NC1CCCCC1F C(=O)(C(CCC(N)=O)N(C)C)N1CCCC(CNC(C(CC(=O)OC)C)=O)CC1 C(=O)(N(OC)C(C)CC)C1CCN(C(C2CC(CCC)C2)=O)CC1O c1(C(=O)NC2CN(C(CC(OCC)OC)=O)CC(O)C2)cncc2c1CCCC2 C(C(CC(F)(F)F)NC(c1cc[nH]c1C)=O)NC(C(COC)(F)F)=O c1(OC)cc(F)cc(F)c1.c1(NC(=O)O)cccc(CC2CC(NC(C)(C)C)CC2O)c1 N#CC1(Nc2cc(Oc3ccccc3)ns2)CCN(C(=O)NCc2ccco2)C1 N#Cc1cc(F)c(C(=O)NCC2CCCCC2NC(=O)CCC2CCC2)c(F)c1 CCCC(CC)CC(=O)N1CCOC(CNC(=O)C=Cc2cccc(C#N)c2)C1 C1(NC(COC(C)C)=O)CC2CC(NC(=O)C(C)(C)C3(O)CCOC3)CC12 C1(CCCn2c(N(CCOC)C)nnc2Cc2ncnn2C)CCC(F)(F)CC1.OC C(C(C(=O)NC1CCOC1)N(C(CC)CC)C)(c1cn[nH]c1)OCC c1(C(=O)NC2C(C(N3CCC(C#N)C3)=O)C2)cc(Cl)cc(Cl)c1Cl C(=O)(CCCC(=C)C)NCC1(C(N2CCN(CC#C)CC2)=O)CC1 CCCC(CCCS(C)(=O)=O)C(=O)NC1CC(NC(c2ccc(CO)o2)=O)C1 CCC(CC(C)C)C(=O)NC12CCC(CNC(c3cnc(C)cn3)=O)(CC1)OC2 c1(C(N2CC(NC(C3C(COC)C3)=O)C(O)C2)=O)ccc2c(c1)NC(=O)C(C)S2 N1(C(CC(C)(C)C#N)=O)CCC(C2CC(NC(C3(C)CC4(CC4)C3)=O)C2)C1 c1(CC(=O)NCC=CC2N(C(C=CC=CC)=O)CCC2)cccc2c1OCO2 N1(C(c2scc(C)c2)=O)CC2CC(NC(=O)Cc3cccc(C)c3Cl)C1C2 C(=O)(C(C)(C)CS(C)(=O)=O)N1CCN(C(c2ccc(C=C)cc2)=O)C(C)C1 Cc1cc(C(N2CCCC(C)(C(=O)NCc3c(C)nn(C)c3C)C2)=O)cc(C)n1 CC(C)CC(C)(C)C(=O)N1CCCC(C(C)NC(c2cnc3ccnn3c2)=O)C1 C1(CC)CN(C(C2(C(=O)NC3CCC(Cn4ccnc4)O3)CC2)=O)CCN1C N1(C(CCCOCC=C)=O)CC(C)CN(C(c2sccc2OC)=O)C(C)C1 C(=O)(C(F)(F)CCn1cccn1)NCC1C2CN(C(C(CCC)N(C)C)=O)CC21 C(=O)(C1=C(C)C(C)(C)OC1=O)NCCC(CC)(CC)NC(CC(C=C)CCC)=O N1(C(c2ncn(CC)c2)=O)CC2CC1CN(C(C1CC3CC1CO3)=O)C2 c1(NC2CCCC(NC(c3cn(C(C)C)nn3)=O)C2)ncnc2ccc(O)cc12 C1(C(=O)NC(C2(C(=O)NCCCC=C)CC2)C)CC=C(C)CC1 N1(CC(N2CC(C)(C(C)C(=O)Nc3cc(Cl)no3)C2)=O)CCC(O)CC1 CN1N=CC(CC(=O)NCC2(C(C)(C)C)CCN(C(=O)CNS(N)(=O)=O)C2)C1=O c1(OC)cc(OC)cc(C(=O)NCC(O)CN(C(=O)CC(O)C(C)C)C)c1 S(=O)(=O)(c1c[nH]c(C(=O)O)c1)NCC1CC(C(F)F)(OC)C1 c1(NC(C2CN(C(c3ccc(Br)o3)=O)C2)=O)cc(F)ccc1[N+](=O)[O-] C1(CCNC(=O)C(O)C2CCCC2)CCCN(C(=O)Cc2cc[nH]c2)C1 CC1CC(NC(=O)CN2CCCCCC2)CN1C(=O)CN1CCCCC1=O C(=O)(C1=CCOCC1)NC(C1(CNC(c2cncn2C)=O)CC1)C O=C(C1=CCCS1)NCc1cccc(CNC(C2CCCS2)=O)c1 N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CCC(NC(=O)C=CCO)C(C)(C)C1 C(=O)(CS(=O)(=O)N(C)C)N(C1CCN(C(CCN(CCCCC)C)=O)C1)C N1(C(C(CCC)CC)=O)CCC2C(CCN2C(c2ccc(C)c(C)n2)=O)C1 c1(C(=O)NCC=CC(=O)NOCCCF)cc2n(n1)CCO2.C1(CO)CCCC1 C(=O)(CC(F)(F)C(F)(F)F)NCC1CCN(C(c2cc(CCC)c(Cl)cc2)=O)C1 C1(C(N2CCCN(C(CC3CC(=C)C3)=O)CC2C)=O)CCOC2(CCCCC2)C1 Cc1c[nH]c(C(=O)N(C2CC2)CC2CCCN2C(C2CNC(=O)C2)=O)c1 Cc1cc([N+](=O)[O-])c(NC(c2ncc(-c3cnc(O)nc3O)cn2)=O)cc1C c1(N(C(CCCOC)C)C)cc(NCC(C)C(F)(F)F)ncn1 N1(C(C2(C)OCCO2)=O)CC2CC1C2C(=O)NC1CCC(F)(F)C1 C1(CNC(COC(C)C)=O)CN2CCCCC2CN1C(=O)CCc1nccn1C C=CCC(CNC(C1(OC)CCC(C)C1)=O)C(=O)NC1CCC(N(C)C)C1 C1(C(=O)NC2(C)CN(C(C3(n4cccn4)CCCC3)=O)C2)COC2(CO)CC1C2 C1(C(=O)NC(c2ncnn2C)CC)CC2(CCC2)CN1C(c1n[nH]c(C)c1C)=O c1(CN2C(=O)CN(C(=O)OC(C)(C)C)C2)ccccc1N1CCOCC1 N1(C(CNC(N)=O)=O)CCN(Cc2cc(Br)c[nH]2)C2CC12 CCCC(C)CC(=O)N1CC(C)(C)CC1CC(=O)NCC(O)CF C1(NC(CC(CC)NC(C2(O)CCC2)=O)=O)CC2COCC(C1)C2 C12(O)CCCN(C1)C(=O)C(O)CN2.C1(C(=O)OC(C)(C)C)CCN1CN(C)C C1(CC(N)=O)CN(C(C2C=CCN2C(C2C3COCC23)=O)=O)CCO1 C(C(=O)NC(C1CC(NC(C2CC=CC2)=O)C1)C)(C(C)(C)C)SC N1(C(C2(CC#C)CC=CCC2)=O)CCCN(C(=O)C(O)COC)CC1 C1(CS(=O)(=O)NCC(=O)OC(C)(C)C)C(=O)NCCN1c1ccc(C(F)F)cc1 c1(N(CCCNC(CC(C)C2CC2)=O)C)cc(Cl)nc(C(C)(C)C)n1 C1(OC)CN(C(=O)CCCN(C)C(c2ccn(C3CC3(F)F)n2)=O)CC1OC c1(OC)ccc(COC(C(c2sccc2C)N(C)C(C)C2CC2)=O)cc1OC C(c1cccc2cccnc12)=CC(N1C2CN(C(CC=CCC)=O)C(CC2)C1)=O C1(NC(c2cc(COC)cn2C)=O)CN(C(c2ccc(F)c(C)c2)=O)CCC1F N(S(=O)(=O)N(C)C)CC(=O)N(CC)CC1CCCN1C(=O)CC1CCCC1 C12CCCCN1C(=O)N2.c1(NC(COC)C2CC2)cc(OC(C)(C)C)ccn1 N1(C(Cn2c(C)ccn2)=O)CCC(C)C(CNC(c2ccc(C3CC3)s2)=O)C1 CC1CN(C(c2cn[nH]c2)=O)CCN1C(c1cc(O)cc(O)c1)=O C1(NC(=O)COCCF)CCC(CNC(=O)C2CC2)C1 CC1CCCC=C1C(=O)NC1CCN(C(=O)CCc2nc[nH]n2)CC1CO c1(C(=O)NCC(n2cc(CC3CCCN(C)C3)nn2)C)ccc(C2CC2)cc1 c1(C(=O)NC2CN(C(C3C(C(=O)OC)CC3)=O)CC2O)cc2nc(F)ccc2o1 C=CCC(CC)C(=O)N1CCC(N(C(C2CC3CCC2CC3)=O)CC)C1 c1(C(=O)NCC(CN(C(CNC(CC)=O)=O)C)C)cn(C)c2ccc(F)cc12 C1(CC)(CC)CC(C(N2CCCC2CC(=O)NC(C)C(C)n2cccn2)=O)C1 Cc1ccc(Cl)c(F)c1C(=O)NC1CCN(C(=O)Cn2ncccc2=O)C1 c1(CNC(c2nc(COC)sc2)(C)C)cccc(C)c1F CCCC(CC)CC(=O)NC1CN(c2cc(C(N)=O)nc(Cl)n2)CC1(C)C c1(C(=O)NC(C2OCCN(c3nccc(OC)n3)C2)C)c(Cl)oc2ccccc12 C1(CC(=O)NC2C(C(=O)OC)CC2)CCCN1NC(=O)CN1CSCC1=O c1(C(=O)NCc2ccccc2CNC(C2CC=CCC2)=O)cnc2[nH]ncc2c1 O(N1CCC(NC(=O)C(C(C)C)NC(C2CCCC(CF)C2)=O)CC1)CC C(C(C)C(F)C(=O)N1CC2C(C)C2C1)NC(CN1C(C)CCC1)=O C(C(=O)N(CCC(=O)NC1CCN2CCCC12)OC)c1ncc(CC)nc1 C(=O)(C(C)C(O)C(C)C)N(C(C)CNC(c1cn(CC(N)=O)nn1)=O)CC CC(C)C(C(=O)N(C1CCC(NC(=O)CCN2CCC2)CC1)C)C1CCC1 C1(N(C)C(c2cccs2)=O)CN(C(c2cc(N)cnc2Cl)=O)CC12CC2 N1(C(=O)CCNCC2(O)CNC2)CC(c2ccccc2)CC1=O O=C(C1=C(Cl)CC1)NC1CCCC1CNC(c1cnn[nH]1)=O N1(C(c2cc(CC)oc2C)=O)CC2(CCC(Nc3cc(C)ncn3)CC2)C1 C12(C(N3C(C(C)NC(=O)C(c4ccccc4)F)CCC3)=O)CC(C)(CCO1)C2 C(c1ccc(C(N)=O)o1)=CC(=O)NC(CNC(CC1(OCC)CCC1)=O)(C)CO C#Cc1ccc(C(N2CCN(C(c3cc(CCC)n(C)n3)=O)C(C)C2)=O)cc1 CC.C(COCCN)=CC.C1CN(C)CCN1.C(CO)OCCO c1(N(CCOC)C)nc2ccc(NCCCOC)cc2c(=NCC(=O)O)[nH]1 C1(NC(C(C2CC2)OCC)=O)CC2CCC1N2C(c1ccc(C)c(C(C)=O)c1)=O c1(C(N2CCCCC2c2ccco2)C(=O)NCC=C)ccc(F)cc1Cl c1(C(N(CCCNC(C2(CC)COC2)=O)C)=O)cccc2c1CCOC2 c1(C(=O)NCC2CCN(C(c3nccc(C)c3)=O)C2)c(F)ccnc1F Cc1cnc(C#N)c(N(C(c2cncc(-c3ccc(Cl)c(F)c3F)n2)=O)c2cccs2)n1 C1(C(N2CCC(C(=O)OC)C2)=O)CCCN(C(c2cccc(CC#N)c2)=O)C1 C1(NC(C(C(C)O)C)=O)CN(C(C2CC(F)(F)C2)=O)CCC12CCC2 C(C(C)(CC(C)C)NC(c1cc(C2CC2)no1)=O)NC(C(C)(C)OC(C)=O)=O c1(C(C)=O)ccc(C(=O)NC2CC(NC(C3(N=[N+]=[N-])CC3)=O)C(O)C2)cc1C c1(C(=O)NCCN(C(C2(CC=C)CC2)=O)C2CC2)ccc(C#N)cc1C c1(OC)ccc(OC(C)C(N2CCC(CN(C)C(C34CSC(C3)C4)=O)C2)=O)cc1 N1(C(c2c(CNC(Cn3ncc(C)c3)=O)ocn2)=O)CCN(C)CC(C)C1 C12(C(=O)NC(COC)C(=O)O)CCC(C(=O)NS(=O)(=O)c3cccs3)(CC1)CC2 c1(OC)ccc(Cl)c(CN2CCN(C(c3cnc(N(C)C)o3)=O)CC2C(C)C)c1 N1(C(CSc2nc(C)[nH]n2)=O)CC(NC(c2ncccc2C(C)(C)C)=O)C(C)C1 c1(C(=O)OC)cc(OC(C2CC2CC(=O)OC)=O)cc(F)c1 N1(C(Cn2c(CC)ncc2)C)CCC(C(=O)NC(C)C)CC1 n1(CC(C)(C)OC(=O)CCC2COC(=O)O2)ccc2ccccc2c1=O C(CC(C)C)(C(=O)N1CCC(C(=O)NCCCC(O)CO)C(O)C1)OC Cc1cc(-c2csc(NC(c3cccc(C)c3C)=O)c2)cnc1O c1(NC(C2C(C)=CCC=C2)=O)ccc(=NCc2cc(-c3ccccc3)no2)[nH]c1 C1(C(=O)NC(CNC(C=CCOC)=O)(C)CC(C)C)CCC12CCOCC2 C1(c2n(CC(F)F)nnn2)(NC(c2csnn2)C2CC2)CC2(CSC2)C1 c12ccc(cc1Br)[nH]c2=O.c1(C(=O)NCCNC(=O)C2CC2)ccc(I)cc1 C1(CNC(C2CCC(SCC)CC2)=O)CCC(C)N(C(=O)CN(C2CCC2)C)C1 N1(C(c2cc(CC(C)C)no2)C(=O)NCC)CCN(C)CC1CC c1(C(=O)NCc2c(CCNC(c3c(C)cccc3)=O)ocn2)cnn2ccsc12 c1(C(N(CCOC)C(C)C)=O)sc(N2CCC(CC(N)=O)C2)nc1C Cc1nc(=NC2CCC3CN(C(=O)CCc4ncc[nH]4)CC3C2)s[nH]1 Cc1nc(NCc2cc(C)on2)cc(N2CCC(Cl)=C(Cl)C2)n1 N1(C(C2(CC)CCCN2C(=O)CC2CCOC2C)=O)CCCCCCC1C CCC(CC)CC(=O)NCC1CN(C)CCN1C(c1ccc(C2CC2)o1)=O c1(SC)ncc(C(=O)NC2CCC(NC(c3cc(I)ccc3Br)=O)C2)c(Cl)n1 C1(C(=O)NCCCC=CC)CC(NC(=O)CCC(=O)N(C)C)C1(C)C N1(C(C2CNC(=O)O2)=O)CCC(F)(CNC(=O)C(F)(F)c2nccs2)CC1 c1(N(C)C)ncc(C(=O)NC2CCN(C(=O)Cc3ccc(O)cn3)CC2)cc1Cl c12ccc(cc1)C(=O)N1CC(C1)N(C)C(=O)C(C)CS2.CC(=O)OCCO N1(C(C(C(CC)C)N(C)C(c2ccc(N(C)C)nn2)=O)=O)CC2(CCC2(C)C)C1 N1(C(C2C(C(C)(C)O)C2)=O)CCN(C(=O)CC(F)(F)F)C(CC(C)(C)C)C1 CC1COCC(CNC(=O)CC2CCCN2C(=O)COc2ccn(C)n2)O1 c1(C(=O)OC)cc(C(=O)NC(C)CN(C)C(C2C=CC=CC=C2)=O)c(C)s1 N1(C(CCNS(CC)(=O)=O)=O)CCN(C(=O)CC(C)COC)CC1CCO O=C(CCCC(F)(F)F)NCC1CN(C(C2CC23CC(F)(F)C3)=O)CC1O c1(C(N(CCN(C)C(C2CCNC(=O)C2)=O)C)=O)cnc2n(c1=O)CCCCC2 c1(C(=O)OCC)ccc(C(=O)NC2COCC2NC(C23CC(CC2)C3)=O)cc1 C(CC1CC1)(CC(=O)NCc1ccco1)NC(=O)Cc1ccccc1 N1(S(CCc2c(OC)ccc(Br)c2)(=O)=O)CCOC2(C1)CN(C(C)C)C2 CC1(C)CN(C(C2(c3ccc(F)cc3)CCCC2)=O)CC1NC(c1cn[nH]c1)=O c1(OC)cccc(O)c1C(=O)NC1CC(N(C(=O)CCC2(C)CC2)C)C1 C1(OC)CN(C(C2CCSC2)=O)CC1NC(=O)CC1COC(=O)C1 N1(C(c2cc(OC)nn2C)=O)CC(NC(c2c[nH]cc2C(C)(C)C)=O)CC(C)C1 C1(C(=O)NC(C2CCC(C)O2)=O)CC(C2CC2)=NO1.c12cccc(n1)CCCS2 C(=O)(CCC(Cc1ccccc1)n1cnnc1)N(C)C.N12CCC(C1)C2=O Cc1noc(C(C)C)c1C(=O)NC1CCCC1CNC(=O)CN(C)C1CC1 c1(C(C)(C)C)cc(N2CCC(CCNC(C3(C)CC3(F)Cl)=O)C2)ncn1 N1(C(=O)CN2CC3C=CC2C3)CCN(C(c2cc(O)c(O)c(O)c2)=O)CC(O)C1 c1(SC)c(C(=O)NCC(C)CN(C)C(c2ccc(C(C)F)cc2)=O)cnn1C N1(C(C(CCC)C)=O)CC(C(=O)NCC2CCC=CO2)C(C2CC2)C1 c1(NC(c2c(C)cccc2)C)nc(=NCCC(C)F)[nH]c2c(C)nn(C)c12 C1(CC(=O)NCCN(CCCCCC)C(=O)Cn2cc(CO)nn2)CCCCCO1 C(=O)(CCC(C)(F)F)N1CCCC(C(C)NC(c2cc(C)n(C)c2)=O)C1 C(=O)(C1COc2ccccc21)N(CCN(C)C(C1CCC(c2cc[nH]n2)O1)=O)C c1(C(=O)NCC(CC=C)NC(c2ccccc2F)=O)ccc(N)c(F)c1Br Cc1ccc(C(C)N(C)C(c2c(C)n[nH]c2C)=O)cc1 C1(NC(c2c(CC)occ2)=O)CCN(C(=O)C(n2ccc(C3CC3)n2)C)C(C)C1 CCC(C)CC(=O)C(=O)N1C(C(=O)NC2CCC23CCCC3)CCC1C1CC1 Cc1cn2c(C(=O)N(CCNC(=O)C(C)NC(N)=O)C(C)C)cnc2s1 c1(C(N(C(C)CN(C(=O)C=C(Cl)Cl)C)C)=O)cc(C(N)=O)ccn1 CC(C)(F)CCC(=O)N1CCC(CNC(c2cc(Cl)ccc2Br)=O)CC1 C1(=O)C(F)C(C)CN(CC)C2CCN1CC2.C1(=O)CC(=O)N1.CCS.CC c1(CC)scnc1C(=O)NCC(O)CNC(=O)C(c1ccccc1)NC(N)=O c1(OC(C(=O)NC2CCN(C(C3CCOC3)=O)CC2)(F)F)ccc(Cl)c(F)c1 CC(CNC(=O)CC1CCCCC1NC(C1CC(N(C)C)C1)=O)S(C)(=O)=O C1(NC(c2ccnc(C)n2)=O)COC2(CCN(C(c3cc(C)sc3N)=O)C2)C1 CC1=C(C(=O)NCC2CCCC2C(=O)NC(C)(C)CC2CCCC2)CCCO1 C1(NC(c2c(CC)noc2)=O)CN(C(c2cc(C3CC3)on2)=O)C2(CCC2)C1 Cc1cc(C(=O)NC2(CNC(C3CC3F)=O)CC2)ncc1C(F)F C=CC1(C(N2CC(NC(=O)CCc3scnc3C)CC(F)C2)=O)CCCCC1 S(=O)(=O)(c1[nH]c(=NCCC2CC2(Cl)Cl)ccc1Br)NC1S(=O)(=O)CCC1 C=C(C)C(C)(O)C(=O)NCC(C)N(C(c1ccc(C(F)(F)F)cc1)=O)CC Cc1c(F)ccc(C(N2CC3CC(C2)N3C(=O)C2=NOC(C)(C)C2)=O)c1F N1(C(c2nc(CC)oc2)=O)CC2(CCN(C(C3CCN(C)C3)=O)CC2)CC1C c1(CC)cccc(-c2cn(C(C)C(C)C)nn2)c1Cl.C(C(C)C)N N1(C(C(C)OCC2CC2)=O)CC(C(=O)Nc2cc(C#N)ccc2O)CCC1(C)C O=C1COCC2(CNC(c3n[nH]c(CC(F)(F)F)n3)=O)COCCN12 N1(C(C(C(C)C)C2CCC2)=O)CC(CNC(C2(C)CCN(C)CC2)=O)C(C)(C)C1 N1(C(C(C)CC(N)=O)=O)CCCN(C(=O)C(O)C(F)F)CCC1 N1(c2c(C)c(NCCCCN3CCCC3)ncn2)Cc2cccn2C(C)C1 c1(COC)c(NC(C2CN(C(c3ncsc3NC)=O)CCO2)=O)cccc1F c1(OC)ccc(OC(C)C(=O)NCC2(C(F)F)CCN(C(=O)C(C)CO)C2)cc1 Fc1cccc(-n2cc(SCCNC3CCCCCC3)nn2)c1 N1(C(COCCCC)=O)CC2CCCC2(C(=O)NCCc2cnnn2C)C1 C1(NC(c2cnn(C(C)C)n2)=O)CCC(C(N2CC3C=CC3C2)=O)CC1 C1(CNC(=O)NCCc2cc(OCC)ncc2)CC(OC)C12CCC2 c1(CCN2CCC(Cc3n(CC)nnn3)CC2C)cc(C)c(Cl)cc1F N1(C(C23C(C)OC(CO)(C2)C3)=O)CCOC2(C1)CN(C(=O)C(C)CN(C)C)C2 c1(C(N(C2CCCN(C(C3(F)CC3)=O)C2)CC)=O)cnc2c(c1)NC(=O)CS2 c1(CC)cc(=NC(=O)CC2CCCN2C(c2ccc(I)nc2)=O)[nH][nH]1 c1(OC)ccc(CC(C)C(=O)NC2(NC(=O)CNC(=O)CC(C)(C)C)CC2)cc1 CC(C)C(F)C(=O)NCCC1CCCN(C(c2ccc(Cl)cc2)=O)C1 c1(C(N2CC(C(C)NC(=O)CCN3CCCCC3)C2)=O)csc2c(F)cccc12 Cc1nc(C(=O)NC2CC(NC(C3CC4CCC4C3)=O)C2)c2ccnc-2[nH]1 c1(C(=O)NCC(CCNC(C2CC=CC(O)C2)=O)OC)nn(C)c(=O)n1C N1(CCCC=C)CC=C(CCNC(C2CC2c2ccc(F)cc2C)=O)CC1 CCCCCCCC(=O)NC1CC12CCN(C(=O)CC(=O)OCC)CC2 O=C(C1CCCc2ncccc21)NC1C=CCN(C(c2cccnc2O)=O)C1 c1(OC(C)C)ccccc1-c1cn(CC(=O)NCC(c2cccs2)O)nn1 C12(C(=O)NC3CC(CSC)C3)CCC(CC1)N(C(=O)CC1NC(=O)NC1=O)C2 N1(C(C(COC)N(C)C)=O)CCC(O)(CNC(c2ccc(O)nn2)=O)C1 N1(C(C(=O)NCCOC)=O)CCCC12CCN(C(C1CC=CCC1)=O)C2 C1(NC(CC(C(C)C)O)=O)CN(C(C2CCC(C)O2)=O)CC2(CC2)C1 c1(C(=O)NCC2(O)CCN(C(C3(C)C(C)CCC3)=O)CC2)csc(S(N)(=O)=O)c1 C(=O)(C(C)CS(C)(=O)=O)NCCN(C(C(c1ccc(Cl)cc1)CC)=O)C1CCCC1 C(C(C)(C)C#N)N(C)C(=O)NCC1CCCC1c1nc(S)n[nH]1 C1(C)(NC(c2cc(C)ns2)=O)CCCCC1C(=O)NCc1cnccn1 C1(CN(C(=O)C(C2CCCC2)Sc2nc[nH]n2)CCC)CCN(C(=O)COC)C1 Cc1ccc(C(=O)N(C2CCN(c3ccc(F)cc3)C2=O)C)c2ncccc12 N1(C(N2CCC(C)CC2)=O)CCCN(CC2CCOC2)CC1.c12ccc(o1)[nH]c2=O C=C(C)CC(C(=O)N1CC(CC(N2CC(F)CC2CO)=O)C(C)C1)OC c12ccc(F)c(c1)NC2=O.c1(OC)cccc(CC2(CS(C)(=O)=O)CC2)c1 CC1C=C(C(=O)NC2(C)CC(NC(=O)CCP(C)(C)=O)C2)CC1 c1(C(N2CC(OC)(CNC(=O)C(C)(O)C3CCOC3)C2)=O)ccnnc1C c1(CCC(=O)NC2CCN(C(c3nnc(C)s3)=O)C2)c(C)nn(C)c1C CC(C)C(O)CC(=O)NCCC(C)(C)CNC(c1ocnc1C1CC1)=O c1(C(c2ccccc2)C(C)C(=O)NC(c2ccc(Cl)s2)C(=O)OC)nncn1C N1(C(c2cc(CNC(CCCC)=O)oc2)=O)CCN2C(=O)CCC2C1 C1(NC(CC(CCC)O)=O)CCC2(CC1)CCN(C(c1cnn(C)c1CC)=O)C2 C1(NC(C(c2n(C)ncc2)O)=O)CCC(NC(c2cnccn2)=O)CC1 c1(CC(=O)OC)ccc(S(=O)(=O)N2CCN(C(=O)C(C)(C)C)CC(CO)C2)cc1 C(=O)(C#CC1CCOC1)NC1CC2(C(NC(C=Cc3cn(C)nc3)=O)C2)C1 c1(CNC(C2C(n3cc(CCC(C)(C)O)nn3)COC2)=O)nc2cccnc2s1 C1(CC(N2CC(O)(COC)C2)=O)CC2(C1)CN(C(=O)Cc1ccn(C)n1)C2 c1(C(N2CC3C(CNC(C4ON=C(CC)C4)=O)(C3)C2)=O)cnc2[nH]c(O)nc2c1 c1(CC)cnccc1C(=O)NC(C)C(C)NC(=O)C1=CCSC1 CCCCCCCCCCC(=O)N(C)CC1(NC(C2COCC(C)(C)O2)=O)CC1 c1(C(NOCC(=O)OCC)=O)coc2c1CN(C(C1CNC(=O)N1)=O)C2 N1(C(=O)Cc2cccc(C(F)(F)F)c2)CCC(CO)C(NC(=O)C(F)(F)CO)C1 N1(C(C2(OCC)CC2)=O)CCC(C)(CC(=O)NCC2(O)CCC(C)C2)C1 c1(C(=O)NC(C(=O)NC(C)Cn2cccn2)CC2CC2)cc(F)ccc1O c1(C(N2CCC(NC(c3c(Cl)cnc(C)n3)=O)C(C)C2)=O)cnn2ccccc12 c1(C(N(C(C)CCNC(c2cnoc2C2CC2)=O)C)=O)cnc2ccc(F)cn12 C(=O)(C#CC1CCOC1)N(CCNC(C(C)Oc1ccc(F)c(F)c1)=O)C1CC1 C=C(C)CCCC(=O)N1CCCC1CN(C(=O)Cc1c(C)cnn1C)CC Cc1cc(=NCCc2ccsc2)[nH]c(N(C)Cc2ccnn2C(C)C)n1 c1(C(=O)NC2CC(NC(c3ccnc(C)n3)=O)C2)ccc(N)cc1F C12CN(CC1C)C2=O.C1(n2cc(-c3cc(CC)no3)nn2)CCOCC1O c1(OCC)ccc(C)cc1CC(N1CC(NC(=O)C(CCSC)NC=O)C1)=O N1(C(COCC(=C)C)=O)CC(CC(=O)N(CCCN2CC=CC2)CC(C)C)CC1C CC(C)CC(CNC(C1CC(=O)CN1C(=O)CC1CCCOCC1)=O)CO C(=O)(C#CC(C)(C)CNC(=O)C(C)C(=O)OC)NCC#CCC c1(OC(C)C(N2CCC(NC(c3cccnc3O)=O)C2)=O)ncc[nH]c1=O c1(NC(N(C)Cc2ccc(I)cc2)=O)ccc(F)cc1Br C1(NC(C=C(CC)C)=O)CCSC12CN(C(=O)COCc1cccc(C)c1)C2 C(CCS(N)(=O)=O)c1cn(C(C(=O)N(CC(=O)O)Cc2nnc(C)o2)C)nn1 C1(NC(=O)C(c2cccc(C(F)(F)F)c2)O)CCCC(NC(C2(O)CC2)=O)C1 c1(CNC(C(=C)C)(C)C(=O)O)cnn2c1CCC2.C(C)(C)(C)OC(=O)N CC1CCC(C)C1NC(=O)CC1CC(NC(C2OCCC2C)=O)C1(C)C S(=O)(=O)(CCC(F)(F)F)N1CC(CC(=O)N(CC)Cc2cccc(Br)c2)C1 C1(C(=O)NCCC2N(C(c3cccc(CCC)c3)=O)CCC2)CC(=O)NC(C)C1 C1(F)(CNC(c2nc(C)sc2C)=O)CCN(C(=O)CNC2CCCCC2C)CC1 c1(CC(N2CCN(C(c3cc(Cl)co3)=O)CC2CCO)=O)c[nH]c2ccccc12 c1(C(=O)NC2(C(=O)NC(c3cc(C)on3)C)CC2C)cnc(O)c(F)c1 C(=O)(CS(=O)(=O)CCO)N1CCC(CNC(C2=C(C)OCC2)=O)(CO)C1 Cn1cncc1C(N1CCC(CNc2cnnn2-c2ccccc2)C1)=O C(=O)(C(C)C(C)c1ccc(Cl)cc1)N(CCNC(C1(OC)CCC1)=O)C(C)C C1(CC)C(C(=O)N(C(C)C)CC2CCC2)CCCN1C(=O)CN1CC(=O)NC1=O CCC(CC)(C(=O)NC1CCC1NC(=O)C(O)c1ccco1)c1ccc(Cl)cc1 c1(C(C(=O)NC2CC(N(C(CN(C(C)=O)C)=O)C)C2)C)ccc(Br)cc1 C1(C(=O)NCc2nc(CC)oc2)CC2CCC(C1)N2C(C1CS(=O)(=O)C1)=O C(=O)(C1=NOC(C)C1C)NC1C(NC(c2cccc(CC)n2)=O)COCC1 C1(Nc2c(C#N)cncn2)CCCCCN(C(c2ccc(-c3cc[nH]n3)o2)=O)C1 C1(NC(=O)OC(c2ccc(OC)cc2)C)CCOC(=O)N1.CC(C)(C)O CC(C)(C)CC(CNCc1cn(Cc2ccccc2)nn1)CO c1(C(=O)NCCNC(C(c2cccc(OC)c2)C)=O)ccc([N+](=O)[O-])[nH]1 C1(C)(C(=O)NC(CC)C)CN(C(=O)C=Cc2ccncc2)C(C)(C)C1 C1(C(N(C2CN(C(=O)C(C)(Cl)Cl)CC2F)C)=O)CCCC1(C)O N1(C(C(C)c2cccs2)=O)C(CC(=O)NCC(C)C(C)(F)F)C2CCCC12 C(=O)(C(C)C(C)NC(=O)C#CC(C)C)N(CC(C)C#N)CC C1(CCC)CN(C(c2cnc[nH]c2=N)=O)CCN1C(C1(C(=O)OC)C=CCC1)=O C(=O)(CCCC(C)=O)NC1C(CC)N(C(c2cn(C(F)(F)CO)nn2)=O)CC1 C1(C(=O)OCC)CCN(C(=O)CCCCc2ccc(OCC)cc2)CC1 N1(C(c2cc(C)nn2C)=O)C2CCCC1CN(C(=O)CCCS(C)(=O)=O)CC2 Cc1oc(C2CC2)nc1C(=O)NCC(C)(CO)NC(=O)CCC1CCC(=O)N1 C1(NC(c2ccn(C(C)C)n2)=O)C2CCN(C(c3cc(C(F)F)cs3)=O)C12 N1(C(C(C)SC(C)C)=O)CC2(CNC(=O)Cc3cnc(C4CC4)[nH]3)CCC1CC2 C1(C)(CC(=O)NC(C2CN(C(c3ccoc3C(F)(F)F)=O)C2)C)CCCC1 CC1(C(=O)NCCC2(C(=O)NCC(c3cccs3)O)CCCC2)CC=CC1 C(c1ccc(Cl)cc1)=CC(=O)NCCCCCCN(C(=O)CCn1cccc1)C C1(C(N2CC(F)(CNC(C3CC3C(F)(F)F)=O)C2)=O)CCCOCC1 N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)C(C)N2CCCC2)CC1(C)C CC1(C)CCN(C(=O)COc2ccon2)CC1NC(C1CC2CCC1C2)=O Cc1c(C(=O)NC(C2CN(C(=O)CN3CSCC3=O)CCO2)C)ccn1C1CC1 C1(CC(=O)NCCN2CCN(C(C3(C)CC4CC4C3)=O)CC2)CC(C)(C)OC1=O C(CCCCCNC(C1CC1Cl)=O)NC(CCC1CC(C(=O)OC)C1)=O O(N1CCC(CC(=O)NC2CCN(C(=O)CC3CCC(=O)C3C)CC2)CC1)CC N1(C(C2C(=C)C2)=O)CC(O)CC1CNC(=O)Cc1ccccc1O C=C1CC2(C1)CC(C(N1CC(NC(c3cn(C)nc3C(F)F)=O)CC(O)C1)=O)C2 c1(C(=O)NC2CCCC(CNC(c3ccc(CC)s3)=O)C2)cc2c(nn1)CCC2 Cc1cc(Cl)c(C(N2CCOCC(NC(C3OCCCO3)=O)C2)=O)cc1C CN1CCN(CC(c2ccc(CN3CCCC3(C)CCCO)cc2)=O)CC1 C(C)(C)(C(C)CC(=O)N1CC(C(N)=O)(OC)C1)NC(c1cc(OCC)no1)=O N1(C(C(C)(C(C)C)OC)=O)CC(CO)C2(C1)CN(C(C1(C)CC1C(F)(F)F)=O)C2 C1(NC(C2C(CCC)CN(C(=O)C(CC)OCC)C2)=O)CC(C)CCC1O C1(C(=O)NC(COC)(C)C)CCC(C)(C)N(C(=O)C(C)S(C)(=O)=O)C1 N#Cc1ccc(C(=O)NC2CC2NC(=O)C2=CCCCC2)cc1C(F)(F)F c1(C(N2CCC(CN(C(COCCC=C)=O)C)C2)=O)cncc(N)c1 C1(CNC(CCSCCCC)=O)C(C)CCCN1C(c1ccnn1CCOC)=O C1(C(N2CCN(CCO)CC2)=O)N(C(c2cnsc2)=O)CC12CCCC2 CC(CNC(=O)CC1(O)CCC1)(C1CCC1)NC(C1CC1c1cnc[nH]1)=O N1(C(c2n(C(C)C)ncc2)=O)CCC(O)(CN(C)C(C2CCCN(C)C2)=O)CC1 C(=O)(C(C)N(C(=O)CCOC1CC1)C)N(C(C#C)C)C.C C(CN=c1cc(C)nc(C)[nH]1)C1CC(NC(c2c(COC)cccc2)=O)C1 C1(OCC)(COC)CCN(S(=O)(=O)Cc2noc(-c3ccccc3)n2)C1 c1(C(N(C2CN(C(C(CC=C)(C)C)=O)CC2O)C)=O)ccnc2ccnn12 C1(NC(c2[nH]cc(CC)c2)=O)CCN(C(c2csc(C3CC3)n2)=O)CC1(C)C CC(C)C(O)C(=O)NC1(CNC(c2cc(O)no2)=O)CC1 C(=O)(CCCCC(C)=O)NC(CCNC(C(CCC)OCC)=O)(C)C N1(C(COCCCC#C)=O)CCCC(NC(=O)CCc2nc(CC)no2)C(F)C1 c1(C(=O)NCC2(C)CCCN2C(=O)CC2(O)CCOC2)cccc2sncc12 CCCCCCC(=O)NC(C)CCCCNC(c1nn(C)c(Cl)c1Cl)=O C1(NC(C(CC)C)=O)CCCCC1CNC(c1ccc(C(F)(F)F)nn1)=O N1(CCC)CCC(C(=O)NC2CCN(C(C3(C(F)F)CC3)=O)CC2)CC1 c1(C(=O)NC2CCC(c3cn(C(CC=C)CC)nn3)C2)cc(C#N)ccc1C c1(CC)ccc(F)c(C2CC2)c1.C12CC1(C)CC(=O)N(C1CC1)CCCNC2=O C1(NC(CCSCC(N)=O)=O)CC2CCC1C(NC(C1CC3(C1)CC3(F)F)=O)C2 C1(CNC(C(CC)NC(C)=O)=O)N(C(C2CN3CCC2C3)=O)CCCC1(C)C C1(C(NOCC(=O)NC2CCC(CC3CC3)C2)=O)CCCOC1 Cc1n[nH]c(=NC(C)(C)CC2CCN(C(c3ccc4c(c3)COCC4)=O)CC2)o1 Cc1ccc(OCC(=O)NC2CC3(C2)CC3NC(C2CC3COCC3C2)=O)cc1C N(C(=NCC(F)F)NCC(C)(C)C)CC1C(C)CCC1 c1(CCC(=O)O)nc(C(N2CCC(COCF)C2)=O)cs1 c1(C(N(CCC)CCC)=O)cnc(-c2nc(-c3ccccc3)cs2)cn1 CCCCC(C)(F)C(=O)NC1CN(C(c2ccc(OC)s2)=O)CC(C)(C)C1 N1(C(c2n(C)nc(O)c2)=O)CCN(C(=O)CC2CSCCS2)C(CF)C1 c1(C2C(N(C(=O)NCCCC)CC)CCC2)cccc(Br)c1 c1(C(N2CC(C(=O)NC3CC34CC(O)C4)OCC2)=O)cnc2nccn2c1 c1(NC(CC(CC)C2CC2)=O)cc(Br)c2c(c1)CNCCO2 Cc1nccn1C(C)C(=O)OC(c1cnn(C(C)C)c1)C Cc1cncc(C(N2CC(C(O)C(=O)NC3CC3(C)C)C2)=O)c1 Cc1ccc(CC(c2nnnn2CCC2CC2)NCC23CCCC2C3)c(Cl)c1 C(=O)(C(C)(C)CNC(N)=O)NCCN(C(Cc1ccn(CC(C)C)n1)=O)C c1(C(=O)NCC2CCOC2C(=O)NCC(O)C2CC2)ccoc1C1CC1 c1(CNc2ccc(NC(c3cc[n+]([O-])cc3)=O)cn2)cc(F)c(Br)cc1Cl CC1CCCCCN1C(=O)CC(C)(C)CNC(=O)CCCCNC(N)=O c1(C(=O)NCC(C)CNC(C2CCCCC2O)=O)ccc(-n2cnnc2)cc1 C(C1=NOC2CN(C(C34CSCC3C4)=O)CC12)NC(C1(CC(C)C)CC1)=O C(C(=O)NC1CC(CNC(=O)C(C)(O)Cc2ccccc2)C1)(C(C)C)CNC(C)=O C(=O)(CCCCN(C(=O)CC1CCC(C)O1)C)N(CC(C)SCC)C C(=O)(CC(O)CNC(C1(CCNC(=O)CCc2cn[nH]c2)CCCC1)=O)OC N#Cc1ccc(C(=O)NC(CNC(=O)CCC2CCCO2)C2CC2)cc1Cl Cn1ncc(CNCC2CCCN2Cc2ccccc2)c1Br Cc1c(C(=O)NC2CN(Cc3ccc(F)cc3Br)CC2C#N)cccc1F C1(NC(CC(CC)SC)=O)CCCN(C(=O)COCCOC)CC1 CCCCCCC(C)C(=O)N1CC(OC)CC(NC(c2cc3sccc3s2)=O)C1 C1(C(=O)NC2C3CN(C(CC4(C)CCOCC4)=O)C2C3)CC2(CO1)CC(F)(F)C2 N1(C(c2ccc(CCCC)cc2)=O)CCC(NC(=O)C(C)CCC)C12CCC2 N1(C(c2c(CC)cco2)=O)CCC(C(=O)N(C2CCN(CCO)CC2)C)C1(C)C CCC(CCC(=O)N1CCCCC1CCCNC(=O)CC1(c2ccon2)CC1)OC CC1CN(C(=O)CCC#N)CCN1C(=O)C=CCCCCCOC C1(C(=O)N(CCSC)CC)C2CCC(C2)N1C(=O)CCC1CCCO1 C1(C(N2CCC(NC(CCc3n(C)cnc3)=O)C2)=O)CCCN1C=O C1(NC(=O)CC(C2CC2)C2CC2)CCC(NC(C2CC23CCC3)=O)CC1 N1(C(C2C(C(N)=O)CC2)=O)CC2CCN(C(=O)CCCC3CCCC3)C2C1 c1(C(=O)NCC(CN(C(C(CC)C(=O)OC)=O)C)O)c[nH]c2cccc(C)c12 Cc1cccc(CN2CCC(CNC(c3ccc(F)cn3)=O)C2)n1 Cc1ccc(S(N)(=O)=O)cc1C(=O)NCC(C(C)C)NC(C1(C(F)F)CCC1)=O c1(C(=O)NC2CC(C(=O)Nc3cc(F)c(C)c(Br)c3)C2)cc2cccc(Cl)c2s1 CC1(CNC(C2CCC=CC2NC(=O)C(=C2CCCCC2)F)=O)CC2CC2C1 C1(NC(C(CO)OC)=O)CC(F)CN(C(c2ccnc(CN(C)C)c2)=O)C1 C1(C(=O)NCCCOCCC(=O)NC(C)CC(C)O)CN(C)CCO1 c1(C(=O)NCC(CCCC)NC(=O)CN(C)CC)cc(F)c(OC)cc1Br c1(C(N(CC(C)CNC(C2CCCOC2)=O)C)=O)cc2ccc(F)cc2o1 c1(C(=O)NCc2ncn(C)c2)cc2cccc(-c3ccc(OCC#N)cc3)c2o1 N1(C(c2c(C)cn(C)n2)=O)CCCCCC(NC(=O)Cc2csnc2C)C1 C#CC1(C)CCCN(C(=O)C(C)N(C(=O)C=CCCC)C)C1 C1(NC(c2cccc(C#C)c2C)=O)CN(C(=O)CCCOC(C)=O)C2(CCOC2)C1 CCCC(C(O)C(=O)N1CCCC(C)(CO)C1)NC(C1(CC)CC1)=O C(C(=O)NCC1C=CC(NC(=O)C=CC(c2cccc(C)c2)=O)C1)(C(C)C)SC N1(C(C(CCC)OC)=O)CCN(C(c2ccc(CF)cc2)=O)C(CC2CC2)C1 N1(C(C(C(C)C)O)=O)CC2CCCCC2(NC(c2ccc3c(c2)NC(=O)C3)=O)C1 N(C1CC(=O)c2ccccc21)C(N1CCCC(C(C(=O)OC)O)C1)=O Cc1c(C(=O)NCC(C)CNC(C2CC2F)=O)cncc1F O=C(C#CC1CCCC1)NC1CCC(C(N2CCc3cncnc3C2)=O)CC1 c1(C(N2C(C)CC(NC(c3ccnc(Cl)c3N)=O)C2)=O)ccc(Cl)nc1Cl N1(C(C2(C)CC(C#N)C2)=O)CC2CCN(C(c3n[nH]cc3Br)=O)CC2C1 c1(CNCC(c2ccc(F)cc2)(C)O)cc2cc(Br)cc(F)c2o1 CCC(CCCC(=O)N(C)C(c1cccs1)C)NC1CCCC1 O=S(=O)(c1cccc(Cl)n1)N1CCN(Cc2cc(C(F)(F)F)n[nH]2)C2CC12 C1(CN(C(=O)COCC2CCOC2)C)CCCC(NC(c2ccc(O)cc2)=O)C1 C(=O)(C#CC1CCOCC1)C(C1CC2CN(c3ncc([N+](=O)[O-])cc3F)CC12)=O C(=O)(C(C)(C)CC(=O)OC)NC(C(C(=O)NCC1(CC)CCC(=O)N1)C)C CC1CN(C(=O)CCN2CCP(C)(=O)CC2)CC(C)C1NC(=O)C=CC(C)(C)C c1(CC)cc(C(=O)N(C)CC2C3CN(C(c4oc(CC)cc4C)=O)CC23)ccn1 c1(C(N2CCN(c3cnc4ccnn4c3)CC2)=O)cc([N+](=O)[O-])c2nsnc2c1 N1(C(=O)OC(C)(C)C)CCc2cc(CN3CCC(C)(C)C3CO)ccc2C1 C1(NC(CCC2N(C)CCC2)=O)CN(C(c2cnns2)=O)CCC1F N1(C(C2(C)CC(=C)C2)=O)CCCC(C2CCN(C(C3CCN(C)C3)=O)CC2)C1 N1(C(=O)NC)CCC(C(N2CCC(NC(=O)Cc3ccnn3C3CC3)C2)=O)CC1 CC1(CO)CCN(C(=O)CC2CCN(c3nccc4nccnc34)C2)CC1O C1(O)(C(=O)NCCCN(C(CCNS(C)(=O)=O)=O)CC2CCCC2)CCSCC1 CC(C(=O)NCCN(C)C)=C1CN(C(=O)CC2CCC2)C1 c1(NC(C2C(C(=O)Nc3cnc(OC)c(Br)c3)C2)=O)csc2ccncc12 N1(C(CCOC)=O)CC(NC(=O)CN(c2ncccn2)C)CC12CCCOC2 c1(N2CC(C(C)NC(=O)CSC(F)(F)F)OCC2)ccc([N+](=O)[O-])c(C#N)c1 N1(CCNC(c2c(OC)c[nH]n2)=O)CCN(C(c2scc(C)c2Cl)=O)CC1 c1(CC)ncc(S(=O)(=O)N2CC(C(=O)NCCCO)C2)o1 C(C(C)(C)CN(C(=O)C(C)N(C)C1CC1)C)OC.C12CC1C(=O)CC1(CC1)C(=O)N2 n1(CC(=O)NCC2CC(C)N(C(c3ccc(O)c(N)n3)=O)C2)cc([N+](=O)[O-])cn1 N1(C(c2nc(CC)oc2)=O)CCCN(C(=O)CC2(C#N)CCC2)CC1C C1(C)(c2ccc(C)cc2)NC(=O)N(NC(=O)CC23CC(C(=O)O)C2C3)C1=O S(=O)(=O)(c1cccc(N2CCCC3(CCCC3)C2)n1)N1CC(C)C(C)C1 CN1CCC2CCN(C(C3(NC(=O)CCc4cn[nH]c4)CC(F)(F)C3)=O)CC12 S(=O)(=O)(c1cnn(C)c1)CN.C(=O)(C(N1CCCC1)C1CC1)N(C)CC1(C(=O)N)CC1 Cc1nn(CCO)c(C)c1C(=O)N(C)CCN(C)C(C1CN(C(N)=O)C1)=O C(=O)(CCC(C)(F)F)N1CC(n2cc(CNC(C3CC(C)(CC)C3)=O)nn2)C1 c1(C(=O)NC(C)CC2CN(C(=O)CO)C2)c[nH]c(=N)s1 N1(C(C(COC)N(C)C)=O)CCC(C2(NC(=O)Cc3csc(C)c3)CC2)C1 N1(C(C2CCC2CC2CC2)=O)CCC(n2cccn2)(C(=O)NCC23CC2C3)CC1 CCC(C)(O)C(=O)N1CCC(OCC(=O)NCCSC2CC2)C1.C1C(=O)N1 c1(C(=O)NC2CCCN(C(=O)C(F)CC3CCC3)CC2)ccc(O)c([N+](=O)[O-])c1 CC#CC1CCN(C(C2CN(C(C3CCC(C(=O)OC)C3)=O)CCO2)=O)C1 C(=O)(C(C(C)C)NC(c1n[nH]c(=N)[nH]1)=O)N(CCCC(=O)NC)C Cc1cc(C(=O)NC2CC(C)OC2=O)cc(O)n1 Cc1cc(C(=O)N(CCNC(C2CC3CC3C2)=O)C(C)C)c(F)c(Br)c1 C1(NC(=O)C2=NOCC2)COC2(C1)CN(C(C1(C(=O)NC3CCOC3)CC1)=O)C2 c1(C(N2C(C(=O)OCc3c(OC)nccn3)CSCC2)=O)ccc2c(c1)OCO2 N1(CC2(C(=O)NC(=O)CCCC3CCCO3)CC(=C)C2)CCCN(CC)CC1 C(=O)(C1=CC2CCCC12)NC1(C)CCN(C(Cn2c(C)ccn2)=O)CC1 C(=O)(C1=CC2(CCN(C(c3ccc(CO)s3)=O)C2)C1)N1CC(C(C)(C)C)C1 c1(NC(C(CNC(C2(OC)CCOC2)=O)CC2CCCC2)=O)cc(C)ccc1O C(CN=C(NCC(c1ccncc1)C)NC1CC1C)OCC Cc1ccc2c(c1)C(C(=O)NC(CNC(c1cc(C)c(F)cn1)=O)CO)C2 C(=O)(CCCCCCN=[N+]=[N-])NCC(CC)NC(c1cnn(CC(F)F)n1)=O C#CCCC(O)C(=O)NCC1CC(F)(CNC(C2(CCC=C)CCOCC2)=O)C1 NS(=O)(=O)CCCCCC(=O)N1CC(NC(c2ccc(F)nc2)=O)C1 O(NC(=O)C(F)C(C)C)C(CC(C)C)C(=O)N1CCN(CCF)CC1 C1(NC(C2(C(=O)OC)CC2)=O)C=CCN(C(=O)Cc2cccc(NC(C)=O)c2)C1 C(C(=O)NOCC(F)F)(C1CN(C(c2ccc(C)o2)=O)C1)OC c1(C(=O)NCC(C)N(C(Cc2c(F)ccc(OC)c2)=O)C)ccc2c(c1)NCC2 Cc1cc(C(=O)NC2CN(Cc3ncccc3Cl)CC2C#N)c2cc[nH]c2c1 c1(C(=O)NC(C(C)NC(C2COC(C)C2)=O)CO)c(F)cc(C#N)cc1F C1(NC(CCc2ccc(SC)cc2)=O)CCN(C(c2ccccc2Cl)=O)C12CC2 C1(C(N2CCCC(OCC)C2)=O)CN(C(C2CC3CCCC3C2)=O)CC12CCC2 N12CC(C3(CC3)C1)CCC(=O)NOCC(=O)N(C)CC2=O.C(CCOC)OC c1(NCc2c(C)cc(N)cc2)[nH]c(=NC2CC3CC3C2)nc2sccc12 CC(C(=O)NCC1(C(N2CC(S(N)(=O)=O)C2)=O)CCCO1)C(F)(F)F N1(C(CNC(C2CC2(C)C)=O)C)CCN(C(c2nc(NC(C)=O)sc2)=O)CC1 c1(C(=O)NC(CCCNC(c2c(C)[nH]c(C)c2C)=O)(C)C)cnc2cccnn12 N1(C(C2C(C)(C)CC2)=O)CCC2(C1)CN(C(=O)CC1CCC1)C2 c1(NC(CN2CCC(C)C2)=O)cccc(CNC(=O)CCc2nc[nH]n2)c1 c1(C(C(=O)NC)N(C)Cc2cc(CO)on2)cccc(COCC)c1 C(C#Cc1ccccc1Cl)N(C1CCN(C(c2cccc(Cl)c2)=O)C1)CCO C1(C(=O)NCC2(F)CCCN(C(CSCC)=O)C2)CCC(F)(F)CC1(C)C c1(-c2cn(CCNC(C34COCC(C3)C4)=O)nn2)cc(Br)ccc1 c1(C(N2CC(O)(C(C)NC(c3c(F)ccc(C)c3)=O)C2)=O)n[nH]c2c1CSCC2 N1(C(CC(CNC(C(C)OCOC)=O)C2CCC2)=O)C2CCCC1CC2 c1(C(=O)NC2C3CN(C(C=C(C)C)=O)C2C3)c(O)cc(=O)n2c1COCC2 c1(CC(=O)NC(CNC(C(COCC)C)=O)CO)ccc2nc(O)[nH]c2c1 c1(C(N2CCC(C)(NC(c3nc(N(C)C)oc3)=O)C2)=O)cc(F)cc(Cl)c1N C1(NC(COCCCC(C)C)=O)CN(C(C2(c3cc[nH]n3)CC2)=O)CCC1CO N(C)(C1CCc2ccc(C(=O)OC)cc21)C(N1C(CC=C(CC)C)CCCC1)=O c1(C(=O)NCCC(=O)NCC(CO)NC(c2cc[nH]c2)=O)cc(Cl)ccc1Cl c1(OC)ccc2c(CCC(=O)NC(C)CN(C)CCOC)c[nH]c2c1 C1(CNC(c2c(C)c[nH]n2)=O)CC2(CC2)CN1C(c1cncc(F)c1C)=O C1(C)(CC)CCC(C(=O)NCCCC(C)(C)NC(c2cc(Br)n(C)n2)=O)O1 C1(C(=O)NC2(COC)CC2)CCC(C2CC2)N1C(=O)CCC1CC1(C)C c1(C(=O)NCC(CNC(C(CC)CN(C)C)=O)(C)F)occ2c1CCC2 CCC(C(C)CN(C)C)NC(=O)C=CCN(C)C(C1(C2CC2)CC1)=O C12(NC(C3CCC(N(C)C)C3)=O)CC(C(F)(F)F)C1CN(C(=O)C=CCO)C2 NC1CC2(C1)C(C(N1CCC(CN3CCCCC3=O)CC1)=O)C2(F)F c1(-c2nc(-c3ccc(N4CC(=O)OCC4)cc3)on2)cc(F)cc(Br)c1F C12(C(=O)NC(C)C=CBr)CC(NC(=O)CC3OCCCO3)(C1)C2 C(C(C(C)C)NC(=O)CC1CCCO1)NC(CSC)=O c1(OCC)cc(CN2CCC2(C)C(N2CCC23CCC3)=O)ccc1OC1CC1 N1(C(C2(C(C)(F)F)CC2)=O)CC2CC(NC(C3CCCCC3(F)F)=O)C2C1 Cc1cc(=O)n(C)cc1C(=O)NC1CC2CC(NC(=O)Cn3cc(Cl)cn3)C1C2 Cc1cc(C(=O)NC(C)CCNC(=O)CCNC(c2ccsc2)=O)ncn1 C(=O)(CCCCCc1ccccc1)N(C1CN(C(=O)CC2CCCN2C)C1)C c1(CC)noc(C)c1C(N1CC(CCNC(C2CCS(=O)CC2)=O)C(C)C1)=O C(=O)(CCCC(F)(F)F)N1CC=C(CNC(c2c(C)cnnc2O)=O)CC1 c1(-n2c(C(C3CC34CCC4)NCCOCCC)nnn2)ccccc1C C1(C(=O)NCC(C)(C)Cn2cc(C3CCCCC3)nn2)(OC)CC(C)(C)C1 C1(CC)CN(C(=O)CNC(=O)CCCSC)CCN1C(C1CCC(F)CC1)=O C1(COC)CN(C(C2CC2C(F)(F)F)=O)CCN1C(=O)Cc1nc(C)no1 c1(COC)ccc(CNC(C2(N(C(=O)CNC)N(C)C)CC2)=O)nc1.C1(SC)CCCC1 C1(CC(=O)NCc2ccc(F)nc2F)CN(C(=O)C(=O)NC2CC2)CC2(CC2)C1 C(C(O)CC(F)(F)F)N(C(=O)CCC(=O)NCCOC1CCOC1)C C1(C(=O)NC(C2CCN(C(=O)CN(S(C)(=O)=O)C)C2)C)COCCOC1 n1(CC(=O)NC2C(OC)CN(C(CN(CCC)C)=O)C2)cc(Cl)c(O)nc1=O Cc1noc(C)c1S(=O)(=O)NCC(=O)N(C1CN(C(C2CCCS2)=O)CC1O)C c1(OCC(=O)NC2CCC(C)(CNC(C=C(CCC)C)=O)C2)c(Cl)cccc1Cl Cc1ccn2ncc(C(N3CCC(O)(CNC(C4CCCCC4O)=O)C3)=O)c2n1 C1(CCC)CN(C(=O)Cc2cn(C)nn2)CCN1C(=O)C=Cc1ccccc1 Cc1cc(C)c(C(=O)NC2CCN(Cc3ncccc3Br)CC2F)c(Cl)n1 Cc1cc(N)c(C(=O)NCC(O)CNC(c2ccccc2CC#N)=O)nc1C N1(c2cc(NC(C)CCN3CCCC3)ncn2)CCC(O)C(F)(F)C1 c1(CCC(N2CC3C(CNC(CC(CC)C)=O)(C3)C2)=O)ccc(Cl)cc1F N1(C(c2cccc(CC)n2)C(=O)NCCCC)CCCC(C)(C#N)C1 Cc1oncc1C(=O)NCC1(O)CC(CNC(=O)CCCn2ccnc2C)C1 c1(CNC(C2CCSC2(C)C)c2n(C(CC)C)nnn2)ccc(N(C)C)nc1 C1(CC(=O)NC2C(NC(c3c(Br)cc(C)c(F)c3)=O)C2)CCc2ccccc2C1 C(C)(C)(CCCC(=O)NCc1ccc(C#N)cn1)NC(C(CN(C)C)O)=O C1(NC(Cn2c(C)nc(C)n2)=O)CC(C)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 C1(CNC(=O)CCC2CC2)CC2(C1)CN(C(=O)CN1CSCC1=O)C2 CN1C(=O)CC(C(N2CCN(C(c3ccnnc3O)=O)CC(O)C2)=O)NC1=O Cc1ccc2occ(C(=O)NC3CC(NC(=O)C(F)=C4CCCC4)C3)c2c1 C(=O)(C(O)C(F)(F)F)N1C(CNC(C2CN(C)CCN2C)=O)CC(COC)C1 N1(C(c2ccc(CNC(CCN(CCC)C)=O)s2)=O)CC2CC1(CO)C2 C1(NC(CC(=O)NCC)=O)CN(C(=O)C(=O)NOC)CC1O c1(C(N2CCC(F)(C(=O)NC(COC)COC)C2)=O)cc(OC)cc(Cl)c1 N1(C(CC2CCN(C(c3cccc(OC)c3OC)=O)C2)=O)CCn2ncnc2C1 C1(NC(=O)CO)CN(C(C23COCC(C2)OC3)=O)CCC1O Cc1cccc(C(CNC(=O)CN(c2ccon2)C)NC(c2csc(C)c2)=O)c1 c1(C(=O)OC2C(C)(C)CCCC2)ccccc1S(=O)(=O)NCC1CC1 C1(NC(c2ccc(C(C)C)o2)=O)CCCC(N(C(=O)CC2CCC2)C)C1 c1(C(=O)NCC2CC(OC)CN2C(c2cc(C)oc2C)=O)ccc(C)nc1O N1(C(C)=O)CCC(C(=O)NC(C)(C)CNC(c2coc(O)n2)=O)CC1 C(=O)(C1COc2ccccc21)N(CCC(C)(C)NC(C1CCC2CC2CC1)=O)C Cc1cc(C(N2CC(=O)CC2C(=O)NCc2cccnc2O)=O)cc(C#N)c1 S(=O)(=O)(c1ccccc1C(C)C)N1CC(C(=O)NCCC#CC)OCC1 Cc1ccc(CCC(=O)NC2CC(C)N(C(c3cnnc(C)c3)=O)C2)cc1 S(=O)(=O)(C1CC2(CCC2)C1)NC1C(CCC)CCCC1 O=C1CCC(C(N2CC(c3ccccc3)(NC(c3ccccc3)=O)C2)=O)CCO1 c1(C(N2C(CC(N3CCC(C)(C(C)C)C3)=O)CCC2)=O)c(Cl)cccc1I c1(C(N(CCN(C(CC(C)C2CCCCC2)=O)C)C)=O)cc2cccn2c(O)n1 C#CCC(CO)NC(=O)C=CCN(C)C(C1(N(C)C)CCC1)=O CS(=O)(=O)c1nccc(N2CCN(C(=O)CN3CCCC3)CC(O)C2)c1[N+](=O)[O-] C1(COC(C2C(=C)CC2)=O)CC2(CCO1)CC2 c1(-n2c(CO)nc(SC)n2)ccc(C)c(Br)c1.CC CC1Cc2ccccc2N2C(=O)N(c3ccc(F)c4c3CCC4)C(=O)C12 C1(C)(CC)C=C(C(=O)NC2COC3(CCC3)C2)C1.C1C(F)C(=O)N2CC1C2 C1(C)(C(N(C2CC(C(=O)NCCCC=CCC=C)C2)C)=O)CN2CCC1CC2 C1(NC(C(C)OCCOC)=O)COC2(C1)CN(C(C1COCCOC1)=O)C2 C1(F)(C(=O)NCC2(COC)N(C(c3cccc(OC)n3)=O)CC2)CC2(CCC2)C1 n1(CC=C)c(N(CC)CC)nnc1CCc1ccccc1 n1(CC)cc(Br)cc1C(=O)NCC1(F)CN(C(=O)C(C)c2ccsc2)C1 N1(C(c2cncc(C)n2)=O)CCN(C(=O)C=C(Cl)Cl)CC12CCC2 c1(OC)cnc(F)cc1C(N1CC(NC(C2COC2)=O)C(c2ccccc2)C1)=O c1(C(=O)NCC2CN(C(COCC=C)=O)C3C2C3)ccc2c[nH]nc2c1 c1(C(N(CC(CNC(COCC=C)=O)(C)C)C)=O)c(CC)noc1C CC1(CNC(=O)Cc2cnsc2)CCC(NC(c2occc2C2CC2)=O)CC1 CC1CC(CNC(c2cnc[nH]2)=O)CN1C(=O)Cc1ccsn1 c1(C(N2CCC(N(C(=O)CC3(NC(C)=O)CC3)CC)C2)=O)cc(O)n(C)n1 N1(C(C(F)=C(C)C)=O)CC(O)CCC1C(=O)NCC(C)(C)C(C)(F)F c1(N2CC(N(C)C)C(C)(C)C2)ccncc1S(=O)(=O)NCc1ccnc(Br)c1 c1(NC(C2(C)CN(C(=O)Nc3ccc(OC)cc3)C2)=O)c(F)cc(Cl)cc1F C12(N(C)C(c3ccc(F)cc3F)=O)CCN(C(=O)CCSc3nccn3C)CC1C2 CC1CCCC=C1C(=O)N1CCCC(N(CCO)C(c2cc[nH]c(=N)c2)=O)C1 N1(C(Cc2c(SCC)cccc2)=O)C2CCC1CN(C(c1cc(C)ccn1)=O)C2 N1(C(CCOCCC)=O)CCC2(CC1)CC(C)N(C(=O)COC1CC(F)(F)C1)C2 Cc1ccc(C(=O)NCC(O)CC(=O)NC(C)CC2CCCCC2)c(C)c1 CC(CCS(C)(=O)=O)NC(c1ccc(CN2CCC2)cc1)=O CC(CC(C)NC(=O)CN=S(C)(C)=O)N=c1nc(C(C)(C)C)nc[nH]1 O=C1CCn2nc(C(=O)NCC3CN(Cc4ccnc(Cl)c4)C3)cc2N1 C1(C(=O)NC2(CNC(CC(C(C)C)N(C)C)=O)CCC2)CCCCCN1C C1(CC#C)(C(=O)NCC(CCNC(=O)C=CC(C)C)OC)CCCOC1 c1(-c2cccc(C(C)(C)C)c2)cc(=NC(=O)C(=O)N2CCCC2)[nH][nH]1 C1(CNC(c2n(C(C)C)ccn2)=O)C(C2CC2)CCN1C(c1cnc[nH]1)=O c1(C(=O)NC(CC(C)NC(C=Cc2c(C)ncs2)=O)C)cc(O)nc(O)n1 N1(C(C(C(C)C)CNC(c2cccs2)=O)=O)CCC2(C=CCO2)CC1 c1(C(N(CCOC(c2c(C)nc(C)o2)=O)CC)C)ncnc2ccsc12.C(C)(C)(C)O C1(CNC(=O)CNC(N2CCCC2)=O)CC2(C1)CN(C(=O)CC1CCC(=O)N1)C2 C1(C(=O)NCC2CCN(C(C(N3C(C)COCC3)=O)C)C2)CC2(CCC2O)C1 O=NN1CCCC1C(N1CC(NC(c2csc(-c3ccccn3)n2)=O)C1)=O N1(C(C(C)N(CC)CC)=O)CCC(CN(C)C(c2ncn(C)c2C)=O)CC1 c1(C(=O)NCC2(F)CN(C(c3cnc(CC(C)C)[nH]3)=O)C2)cccc(Cl)c1F C1(NC(=O)CC2CCCOC2)COC2CN(C(c3ncsc3C3CC3)=O)CC12 N1(CC#C)CCN(C(c2c(Br)cnn2C)C(=O)N(CCCF)C2CC2)CC1=O c1(C(C)Nc2c(C)nccc2)ncccc1[N+](=O)[O-] C(C)(C)(C(=O)N1CCCC1CN(C(=O)C(Cl)=CCl)C1CC1)NC(=O)NCC N1(C(CS(CCC)(=O)=O)=O)CCn2ncc(S(C)(=O)=NC(=O)CSC(=N)N)c2C1 C1(CN(C)C(c2ccn(C(C)(C)C)n2)=O)CCCN1C(C1CC1(C)Br)=O c1(C(N(CC)NC(=O)C(=O)NC2(CO)CC2(F)F)=O)cccc2c1nc(O)n2C N1(C(C(CSC)C)=O)CCCC(CCNC(c2cccc(-c3nnco3)c2)=O)C1 N1(C(=O)Cc2ccc(O)cc2)CC2CCN(C(=O)C3=NOC4(CCC4)C3)C(C2)C1 c1(C(N2CCC(n3cc(C(C)NC(C)=O)nn3)C2)=O)ccc(CC)o1 c1(CC(=O)NC2CCCN(C(C3(F)C(C)C3)=O)C2)ccc2nc(O)[nH]c2c1 C1(OC)CN(C(=O)CCc2ccn(C)n2)CC1NC(=O)Cc1c[nH]nc1C c1(CC(=O)NCC(=C2CN(C(CCN(CC)CC)=O)C2)F)cccc(C)c1Cl N1(C(c2c(CC)con2)=O)CC2CCC1CC2NC(c1c[nH]c2nccc-2c1)=O C(=O)(CCCN(C)N=O)NC(CCN(C(c1c(SC)cnn1C)=O)C)C(C)(C)C Cc1n[nH]c(C)c1-c1ccc(C(=O)N(CCNC(=O)Cc2cnco2)C2CC2)s1 c1(C(=O)NC(C(C)NC(=O)CCc2ccco2)C)ccc(COC)s1 C(C(=O)NCC1CN(C(=O)Cc2cc(C3CC3)on2)C1)(C(C)(C)C)SC c1(CC(N2C(CN)CCC(CCC(=O)OCC)C2)=O)cccc2c1OC(C)(C)C2 S(=O)(=O)(C(F)(F)F)Nc1ccc(C(C2CCN(S(=O)(=O)C(F)F)CC2)(C)C)cc1 CCCCCC(C)CC(=O)NCC(C)NC(c1ccncc1)=O Cc1ccc(C2CCCN2CC(C)Cn2ccnc2)cc1 CC1=C(C(=O)NC(C2CCOC2)CNC(c2cnc(O)n2C)=O)COCC1 Cc1nccc(CCNC(C2(NC(=O)CCC3CCC(=O)C3)CC2(C)C)=O)n1 N1(C(Cc2cc(C)nn2C)=O)CC2(C)CC1(C(N1CCC(F)(C#N)C1)=O)C2 Cc1cc(C(N2CCCC(NC(=O)CC(C)O)C2)=O)cnc1C(F)F c1(CC)onc(C)c1C(N1CC2(NC(C3CC3C(C)C)=O)CC1C2)=O c1(N(CCOC)C)ccc(S(=O)(=O)NCc2ccc(OC)c(Br)n2)cc1 C1(C(C)(C)O)CCN(C(C2(CNC(=O)C(O)C3CC3)CC23CCC3)=O)CC1 N(C1c2ccccc2CC1O)C(=O)NCC1C(C)CCO1 C(=O)(CC1=CCCC1)N(CC(C)O)CCNC(C(CCC)OC)=O C(=O)(CCC(F)(F)C(F)(F)F)NCC(C(C)C)NC(c1scc(OC)c1)=O c1(C(=O)NCC(C)N(C(=O)Cc2ccsn2)C)cc(N)ccc1Br C1(N(C(c2c(C)n(C)nc2)=O)C)CCCN(C(C2CC=CCO2)=O)CC1 c1(NC(=O)Nc2cccc3scnc23)nc2c(s1)CC(N1CCCC1)CC2 c1(C(=O)NCC2CCC(NC(c3n(CC)ncn3)=O)C2)cc(C#N)ccn1 C1(CC)CCC(C(=O)NC2CCCC2CN(C(=O)Cn2ccnc2C)C)O1 C(C1(F)CN(C(=O)COCC)C1)NC(C(COCC=C)c1ccccc1)=O C(C)(C(=O)NC(C1CN(C(=O)CSC2CC2)C1)C)OCC=C CC(C)(C)CC(F)C(=O)N1CCCCC1CCNC(=O)CNC(=O)CC(C)(C)C Cc1cccnc1C(N1CC(CNC(c2cnncc2O)=O)C2CC12)=O N1(C(C(C)SC)=O)CC(NC(=O)CCCc2ccc(F)cc2)CC2(CCC2)C1 Cc1ncnc(C)c1C(=O)NCC12CC(CO1)N(C(c1ccnc(CO)n1)=O)C2 N1(C(C(c2ccccc2)OCC)=O)CCN(C(=O)CS(=O)CC)CC1 C=CCC(CC)C(=O)N1CCCC1(C)CNC(C1CCCC(C(C)(C)C)C1)=O C1(CCC)CCCN(CC2CC=CCC2SC)CC1 c1(N(C(C)C)CC)ccc(C(=O)N(C)CCNc2nc(Cl)sc2Br)cc1 C1(C(=O)NC(C)C(C)(C)NC(c2ccc(CF)cc2)=O)CCCC2(CC2)C1 c1(C(=O)OC)ccnc(N(C)CC2CN(C(c3csc(O)n3)=O)CCO2)n1 C1(CNC(C(C(C)C)OC)=O)CN(C(c2cc(C(F)F)nn2C)=O)C2(CCC2)C1 CC(CN=c1[nH]c2c(c(=NCc3cn(C)cn3)[nH]1)SCC2)C1CCC1 O=C1CC(=O)NC(C(=O)NCc2nocc2C(N2CCCCC2CF)=O)C1 CC(CF)CC(=O)NCC1(CNC(=O)CSC2CC2)CCC1 CCC(C)C(C(=O)NCC(C1CCC1)OC)N(C(=O)CCc1csnn1)C N1(C(C(C(=O)OCC)F)=O)C2CCC1CN(C(=O)CCC=Cc1ccccc1)C2 C=CCCCCC(=O)NC(CCC)C(=O)NCC1(C)C=CCCC1 C1(C(=O)Nc2cc(OC)c[nH]2)(CNC(C2C(Cl)(C(=O)OCC)C2)=O)CS(=O)(=O)C1 N1(CC(=O)NCC2CC2C(=O)NCC2CNC(=O)O2)CC(=O)NC1=O c1(C(N(CCCNC(c2cc(C)on2)=O)CC)=O)cnc2c(c1)CCC(=O)N2 C1(CC)C(NC(c2ccc(C3CC3)s2)=O)CCN1C(=O)Cn1nnnc1C1CC1 c1(C(C)CC(=O)N2CCCC2c2cn(C3(S(N)(=O)=O)CC3)nn2)ccccc1F c1(SCC(=O)NC(C2N(C(CSC(C)C)=O)CCC2)(C)C)cccc[n+]1[O-] CN1CCC2(CCN(C(C3(CCNC(=O)Cc4cnns4)CCCC3)=O)C2)C1 N1(C(C2CC2(Cl)Cl)=O)CCCC2C1CCCCN2C(=O)C=Cc1cocn1 C(CC(O)CNC(=O)C(F)=CC1CC1)NC(=O)CCc1ccc[nH]1 N1(C(C2(CC#C)CC2)=O)CC2(CCCC2NC(=O)C=Cc2scnc2C)C1 N1(C(c2ccc(CC)cn2)=O)CC2(CCNC(=O)CSCCOC)CCC1C2 N1(C(C=NOC)=O)CCC(O)(C(C)NC(c2c[nH]cc2C)=O)C1 CCC(CC(C)C)C(=O)NCc1ccccc1CNC(=O)Cn1ccnc1C N1(C(c2occ(C(=O)OC)c2)=O)CCC(N(C(=O)Cn2nnnc2C)CCO)CC1 C(CN=c1nc(N2CC3CC2CC3O)cc[nH]1)c1c(C)n[nH]c1C C1(CN(C(=O)CCCC2CC2)C)CCCN1C(=O)C(C)(C)n1cncn1 c1(OC2(NC(C=CCN(C(CCCOC)=O)C)=O)CCC2)ccc(C)c(C)c1 c1(-c2ccccc2)cc2n(n1)CCCN(CC1CC3CC3N1)C2 CCC(CO)CCNC(C1CC(NC(C2CS(=O)C2)=O)C1(C)C)=O C(=O)(CC1=CCOCC1)NCC(C(=O)NC1COCC1C1CC1)N(C)C CC(C)CCC(=O)NCc1ccoc1C(=O)NC1C(O)CC1O C1(C(=O)NC2(CO)CC(OC)C2)C=CCN(C(C2CCOC(=O)N2)=O)C1 C(=O)(C(C)S(N)(=O)=O)N(CC(C(N1CCC(COC(C)=O)C1)=O)C)C c1(C(=O)NC2CCN(C(C3=CC(C)(C)C3)=O)CC2F)cc(Br)cc(F)c1F C1(C(N2CCC(N(CCC)C(C3CCCO3)=O)C2)=O)CCC(OC)CC1 C1(CNC(C2CC(NC(C3CCC(C)(CC)O3)=O)C2)=O)OCCCC1(C)C CCCC(C(=O)NC1CCC(F)(CNC(C2CN(C)C2)=O)C1)S(N)(=O)=O C1(CC(N2C(CC(=O)NCC(NOCC)=O)CCC2)=O)CC2(CC2)CO1 CCCC(CNC(=O)CC=CC(C)(C)C)NC(c1cnn(CC)c1)=O C(=O)(C(C)CC(C)(C)C)N1CCC(CNC(c2c(C)c(N)ccc2)=O)C(C)C1 C1(C2NCC(S(C)(=O)=O)C2)CCN(Cc2ccco2)CC12CCC2 C1(=CC(=O)NCC2CN(C(C34COCC3C4)=O)CC2O)C2CC3CC(C2)CC1C3 N1(C(CCNC(N)=O)=O)CCC(C(O)CNC(=O)Cn2cnnc2O)CC1 C1(NC(CC2C(C)(C)C2(C)C)=O)CC2CC1CN(C(=O)C(O)C1CCC1)C2 c1(NC(=O)COC2CCCCC2)ccn2nccc2c1.CC1CC2CCN1C2=O c1(C(C(=O)Nc2ccc(Cl)cc2)N(CCCC=C)CC)cccc(Br)c1F c1(C(N(CC(CC)O)C)=O)nc(CNC(C2CCC(C)(C)O2)=O)oc1C c1(OC)cc(C(=O)N(CCCNC(c2ccc(C)nc2)=O)C2CC2)c2c(c1)CCC2 c1(NC(C)=O)ccc(OCC(=O)NCc2cn(C3CCCC3O)nn2)cc1F c1(CC(=O)NCC2(NC(COC(C)(C)C)=O)CCOC2)cccc(F)c1 CC1(C)CCC12CN(C(C1CSCN1C(c1nnc(O)nc1O)=O)=O)C2 C1(C2CCCCCC2)(C(=O)NCCC2(O)CCN(C(C(CC)N(C)C)=O)C2)CC1 c1(C(N2CCC(N(C(c3ncsc3C)=O)CC)C2)=O)noc2c1CC(F)(F)CC2 CN1N=CC(CC(=O)NC(CC2CC2)CC(=O)NCCC[Si](C)(C)C)C1=O c1(C(C)C)cc(C(=O)NC(C)(C)C(=O)NC(C)C)on1.C1(CO)C(=O)N1 N1(C(C2(OC)CCCCC2)=O)CCC(O)C(NC(=O)C#CC(=O)OC(C)(C)C)C1 c1(C(=O)NC(CNC(CN2CCC(C)CC2)=O)CO)cc2c([nH]1)CCC(C)C2 C(CS(=O)(=O)c1ccc([N+](=O)[O-])cc1)NCC1CC(C(=O)OC)C12CCOCC2 C(=O)(CC(=O)OC(C)(C)C)NC(C)CCNC(c1ccns1)=O Cn1cc(C(=O)NCCC2CC(NC(=O)Cc3ncc(Cl)s3)C2)n(C)c1=O N1(C(c2nc(-c3ccc(OC)cc3)sc2)=O)Cc2c(n(C)[nH]c2=N)C1 N1(C(C(CCCC)C)=O)CCC(C2CN(C(=O)CC3CCCCCO3)C2)CC1 c1(CC)cnc(C(=O)NCC(C)(C)CN(C)C(C2CCCCC2OC)=O)cn1 C1(CNC(C2C(OC)(OC)CC2)=O)CC(F)(F)CN1C(C1CCCCC1(C)C)=O C1(C(=O)NC(CNC(C2(CCC)CCC2)=O)(C)C(C)C)Cc2nnc(C)n2C1 C=C(C)C1OCCC1C(=O)NCCNC(=O)C(O)(CC)c1cccc(Cl)c1 CCCC(CC)C(=O)N1CCCC(NC(=O)CCn2cc(C)cn2)CC1 N1(C(C(c2ccccc2)C)=O)CC2CCN(C(=O)CSC3CCOC3=O)C2C1 CC1OC2CCC1(NC(C1(CC)CCCN(C(=O)C=Cc3ccsc3)C1)=O)C2 C1(CNC(CSCCOC)=O)CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 C1(C)(CNC(CC=CC=C)=O)CCN(C(C2CCCN2c2nc(C)cs2)=O)CC1 C(CC(C)C)(C(=O)NCC1CC2CC2C1)N(C)Cc1c(SC)cccc1 C1(C(=O)Nc2cc(OCC#C)ncc2)CCN(c2ncncc2OC)CC1O N1(C(C(C)(C)O)=O)CCC2(C1)CN(C(=O)CC(O)Sc1ccccc1)CCO2 N1(C(c2nc(C(C)=O)sc2)=O)CCC2(CC1)CC2CNC(C1CCCC1(C)C)=O N1(C(C(C(C)C)NC(C)=O)=O)CC=C(CCNC(C2(N(C)C)CCCC2)=O)CC1 Cc1cc(C(N2CCCC2CCC2CCCCN2C(=O)CSC2CC2)=O)ncn1 Cc1nccn1CCNC(=O)C(C)(C1CC1)N(C)C(C1CCC(=O)C1)=O c1(C(C)NC(=O)C(=O)NCCC(F)(F)CO)ncc(Br)cc1C C1(CNC(=O)COCC(F)F)CC2CCCC2N1C(=O)CCN1CCCCCC1 CCC(C)(CNC(c1ccc(CNC(c2cc(C(F)F)[nH]n2)=O)o1)=O)C(C)O Cc1c(C(N2CC=CC2(C)CO)=O)sc2nc(-c3ccccc3)nc(O)c12 N1(C(C(CC)CCOC)=O)CCC2CCC(C1)N2C(c1cc2cnccc2o1)=O N1(C(C2CC(OC)C2)=O)CCC2CC1CN2C(C1CCC2CC1C2(C)C)=O C1(CCNC(C2CCO2)=O)CCCCN1C(=O)COc1ccccn1 c1(C(N(CCNC(c2cccc(CC(C)C)c2)=O)C2CC2)=O)cc2c([nH]1)CCC2 c1(C(N2C(CCN(C(COC)=O)C)CCCC2)=O)ccc2c(c1)N(C)CC2 c1(C(N2CCC(CCNC(C3C(C(N)=O)C3)=O)C2)=O)ccccc1OC(F)(F)F C(=O)(C(CC(C)(C)C)NC(C1COCCO1)=O)N(CC(C)N(C(C)=O)C)C Cc1csc2c(N3CC4CCN(C(=O)Cn5ccnn5)CC4C3)ncnc12 c1(SC)ccc(O)c(C(N2CCC(N(C)C(c3cnc(O)n3C)=O)C2)=O)c1 C(=O)(C(F)C(C)CNC(=O)C(C)c1ccco1)NC(c1cccc(C)n1)C c1(OCC)cc(C(N2CCC(N(C(=O)CN3CCOC3=O)CCO)C2)=O)[nH]n1 c1(C(=O)NCC2C=CCN(C(C=CC(CC)C)=O)C2)ccc(SC)cc1Cl C12CN(CC13CC3)C(=O)C1C=CCN1C(=O)C2.c1(COC)cc(C)cc(F)c1 c1(C(N2CC(O)(C(C)NC(=O)Cc3csnn3)C2)=O)cn(C)ccc1=O C(=O)(CCCS(N)(=O)=O)N1C(NC(=O)C(C(C)(C)C)OC)CC(OC)C1 C1(C(C)C)CCC(C(C)NC(=O)Nc2ccc(OC(C)C)o2)CC1 c1(C(=O)O)cnc(C)nc1C(=O)NC(C(C)CC)C.C12CC1C2.N(C=O)(CC)CC c1(CNC(C2C(C(C)C)C2)=O)ncoc1C1CN(C(=O)CSc2ccccn2)C1 c1(CNC2CC(CNC(=O)CCC(F)(F)F)C2)c(Cl)c[nH]c2nccc1-2 CC(C)C(F)(F)CC(=O)N1CCC1CNC(c1ccc(C(F)F)nc1)=O C12(CNC(C(SC)SC)=O)CC1CN(C(=O)CCOC1CCOC1)C2 CC(C)(C)C(CNC(=O)CCOCc1ccccn1)NC(c1ccc(Cl)nc1)=O C#CCC(C)(C)C(=O)NCCCC(C)NC(C1COCCN1CC)=O c1(C(C(=O)NC2CC(NC(c3cc(CC)[nH]n3)=O)C(O)C2)O)ccc(Cl)cc1Cl N1(C(CNS(CC)(=O)=O)=O)Cc2ccccc2OC2(C1)CN(C(C1(C)CC1)=O)C2 c1(C(N(CCNC(c2c(CCC)occ2)=O)CCC)=O)ccc2cnccc2c1 c1(CC(=O)NCCN(C(C2(CN(C)C)CC2)=O)C)cnc2ccccc2n1 C1(C(=O)NC2(CNC(C3(CC)CCCCC3)=O)CCCC2)CC2OC(=O)OC2C1 CC1CC(C(=O)NCC2CC(O)CN2C(=O)CC=C(Cl)Cl)c2ccccc2N1 c1(C(=O)NC2CCOCC2NC(C2(O)CC3CCC2C3)=O)ccc([N+](=O)[O-])cn1 N1(C(CSCC#C)=O)CCOCC1CNC(c1cnccc1OC)=O N1(C(C(n2cc(C(C)(C)CO)nn2)C)=O)CCCCC1C(=O)Nc1cnn(C)c1 Cc1n[nH]c2nc(O)c(C(=O)NC3CCC(CSc4ccccc4)CC3)cc12 C(=O)(N=c1cncc(Cl)[nH]1)c1nc(CNC(c2cccnc2)=O)sc1 C(=O)(CCCCCS(C)(=O)=O)N1CCCC(C)(C)C1CNC(=O)C(N)=O C(=O)(C(C)C(C)NC(=O)C(=C1CCCCC1)F)N(C(C(=O)OC)C)C C1(O)(CCNC(c2cc(C(C)(C)C)no2)=O)CCN(C(=O)C2CC2)CC1 c1(C(N2CCCC(NC(C3C(C)C3(F)F)=O)C2)=O)cc2ccccc2cn1 CCC(O)CC(=O)NC12CC1CN(C(=O)Cc1sc(O)nc1O)C2 CC1(CC(=O)NOCC(O)CO)CCCN1C(=O)COCC(F)F N1(C(c2c(F)cc(C)c(F)c2)=O)CCC2(CCN(C(c3nonc3N)=O)CC2)C1 C#CCC(CC(=O)N(C)Cc1cn(C)cn1)NC(=O)CCCN1CCCC1 c1(CN(C(=O)C(=O)NCC2COC(C)(C)O2)CC)ccc(OC)c(OC)c1 C1(NC(CCC(=O)NCC)=O)CCN(C(=O)C(C)n2cnnn2)CC1C C1(CNC(COCCCC(C)C)=O)CN(C(=O)CC2(O)CCOCC2)CC1C c1(C(=O)NCC2(F)CN(C(C(C)CC3CCC3)=O)C2)cnc(O)n(C)c1=O c1(C(=O)NCCOCCNC(C2(CC)CC(F)(F)C2)=O)cnn2c(C)ccnc12 n1(C(C)C(=O)NC2CC(CNC(C3CSC3)=O)C2)cnc2ccccc12 N1(C(CC2CC(=C)C2)=O)CCC2(C1)CN(c1nccnc1F)C2 c1(OC)cccc(S(=O)(=O)Nc2ccc(NC(=O)Cn3cc(Cl)cn3)cc2C)c1 O=C1CC2(CCC2)C(C(N2CC3(CNC(=O)CC4(CO)CC4)CC2CO3)=O)C1 c1(N)ccc(N)c(O)c1.CCC(CC(=O)NCCNC(C(CC)C)=O)c1ccccc1 N1(C(c2c(CC)cnnc2)=O)CC2C=CC1C(C(=O)Nc1cccn(C)c1=O)C2 C1(C(F)(F)F)(NCCNCCCC(=C)C)CC(C)(C)C1 C(C)(CO)(C(=O)N(CCCCN(C(=O)CC(C)n1cccc1)C)C)OC c1(C(=O)NC(C(=O)NCCNC(=O)NC)C2CCOC2)[nH]ccc1C CC1CCN(C(C2COC(=O)N2)=O)CC1NC(c1ncccc1Br)=O C1(C)(C(=O)NCC(C)(C2CC2)NC(=O)Cc2cnoc2)CCCCO1 c1(C(=O)NC2CC2C(=O)Nc2ccccc2O)cccc([N+](=O)[O-])c1 C1(C(N2CC3CC2C3NC(=O)CC2CCSC2)=O)(COC)CCCCO1 c1(NC)cc(Cl)ccc1C(=O)NCC1CC(CNC(=O)C(C2CC2)C2CC2)CO1 C1(C(=O)NCC2(C(N)=O)CN(C(=O)CC3CCCC34CC4)C2)CC2CC(=O)C1O2 c1(C(N2CC(NC(C3CC34CC4)=O)CC3(C2)CC3)=O)cc2cc(F)c(F)cc2[nH]1 N1(C(Cc2c(C)cc(F)cc2)=O)CCCN(C(=O)CCNC(N)=O)CCC1 c1(OC)ccc(OC)c(C(=O)NCC2(O)CCCN(Cc3cccc(O)c3)C2)c1 N1(C(C2(CC)CCC2)=O)CC2(CC(C(=O)NCCCS(C)=O)CO2)C1 c1(C(C)C(=O)NCC2(O)CC(NC(=O)CCc3cscn3)C2)cccc(C#N)c1 N1(C(C(C)NC(CC)=O)=O)C2CCC1CN(C(c1c(Br)cnn1C)=O)C2 CC1OC2(C(N3CC(O)(CCNC(=O)Cn4cc([N+](=O)[O-])cn4)C3)=O)CCC1C2 CCC(CC(=O)NCCN(C(c1nc(NC)oc1C)=O)CC1CC1)SC CC(CC(C)N=c1[nH]c2c(F)cccc2o1)NC(c1cc2c([nH]1)CCC2)=O CCC(C(=O)NC(C)(C)C(C)NC(=O)Cc1ccc(C)o1)NC(N)=O C(CCSC)(C(=O)NCCc1ccn(C)n1)NC(CCCOC)=O C1(C(N2CC(C)C(CNC(C3(C)CC=CCC3)=O)C2)=O)CC2(C1)CC1(CCC1)C2 C=CC1(C(=O)NCC2CC3CCC2N3C(=O)Cn2ccc(=N)[nH]2)CCOCC1 CC1CCN(C(=O)COc2ccc(C#N)cc2)CCN1C(c1nnn(C)n1)=O C(=O)(C(C)S(C)(=O)=O)N1CC2C(NC(c3c(C)[nH]cc3)=O)(C2)C1 CCS(=O)CC(=O)NCCN(C(c1cn(CC(O)CC)nn1)=O)C1CC1 c1(CC)nn(C)cc1C(=O)NCc1cc(C(=O)NOC(C)C(=O)OC)cs1 C1(CS(N2CCCC(Oc3ncccc3Br)C2)(=O)=O)CCNC12CCCC2 C#CCCCCCC(=O)NC(c1ccc(C)cc1)CC(=O)NCCC1CCN(C)C1 c1(C(C)C)[nH]nc(C(N2CC(NC(C3CCC(=O)N3)=O)C(C)C2)=O)c1[N+](=O)[O-] C1(C(N(CCN(C(C)C)C(c2cnccn2)=O)C)=O)OCCN(C)C1=O CC1CC(NC(=O)C(O)CN(C)C)CCN1C(=O)Cc1nc(=N)[nH][nH]1 C#CCC(CC(F)F)NC(=O)C(C)=CCNC(c1ccc(CO)cn1)=O C1(OC)CC(CNC(c2cscc2C(F)F)=O)N(C(=O)C=C(C)c2cccs2)C1 N1(C(C(CC)CO)=O)CC(C2CCCN(C(=O)Cn3cncn3)C2)C1 N1(C(CC2(CNC(=O)CCc3cncs3)CC2)=O)CCc2ccc(F)cc21 C12(C(=O)NC3CC(N(C(CN(C(=O)OC)C)=O)C)C3)CCC(CC(=O)C1)S2(=O)=O N1(CC(C)N(C(c2cnn(CC(F)F)c2)C(=O)NCC2CCC2)C)CCOCC1 c1(C(N(C2CC(NC(C3CCC(OC)CC3)=O)C2)C)=O)ncn2ccc(C)cc12 c1(OC)cc(F)c(C(=O)NC2CCC(C)N(C(=O)C3=C(C)OCCS3)C2)c(F)c1 CCCC(CC)C(=O)N1CC2CC1C2NC(c1ccc(OC)c(C2CC2)n1)=O CCCCC(CNC(c1cc(C)oc1CC)=O)NC(=O)C(C)(C)C1(O)CCOC1 c1(C(=O)OC)cc(CC(N2CCC(NC(=O)C(F)=C(C)C)C(O)C2)=O)ccc1C C1(CNC(C=Cc2ccc(CC)o2)=O)CN(C(=O)Cc2ncc(C)[nH]2)CCCO1 c1(C(N(C)C=O)=O)snnc1C(F)F.C12(CC1)C(=O)NCC(=O)NC2.C1CC1 C1(C2CN(C(c3cc(Cl)ns3)=O)C2)(NC(c2cn(C3COC3)nn2)=O)CC1 CC1CN(C(C2CC3CCC3C2)=O)CC1(C)CNC(=O)COCCN(C)C c1(CC)nc(C)oc1C(N1CCOCC1CN(C)C(c1nccnc1N)=O)=O c1(CC)cccc2c(C(=O)NC(C3CCN(C(=O)CCS(C)=O)CC3)C)c[nH]c12 C12(NC(c3cc(COC)on3)=O)CCCCCC1N(C(c1ccoc1I)=O)CC2 c1(NC(c2c(-c3cccc(OC)c3)cccc2)=O)ccc(P(C)(C)=O)nc1 c1(C(N2CC3(C(C(=O)Nc4c(C#N)nc[nH]4)C3)C2)=O)ccc2nccn2c1 C1(C)(CNC(c2c(CC)sc(=N)[nH]2)=O)CCN(C(=O)C(CC)n2cncn2)CC1 C(=O)(C(N)CS(C)(=O)=O)N(C(c1ccc(C)cc1)c1cn(C)nn1)C1CC1 c1(NC(CSCc2scc(CC)n2)=O)ccc2c(c1)c1ccccc1n2C C1(CNC(CNC(C2CNC(=O)O2)=O)=O)CC2(CCCO2)C1 Cc1nc(NC(C2C3CN(C(c4cccc(Br)c4F)=O)CC23)=O)c(F)c(Cl)n1 C1(C(=O)NC(C2N(C(c3c(C)sc(Cl)n3)=O)CCC2)C)CCCCCCC1 N1(C(c2c(C)noc2C)=O)CCC(NC(c2ccncc2F)=O)C(C(C)C)C1 c1(COCCOC)nccc2c(Br)cccc12.c12cn(nn1)C1CC(C1)NC2=O C=CC(C)(CCOC)C(=O)N1CCN(C(c2cncc(NC)c2)=O)C2(CC2)C1 c1(C(=O)NCC2CC(N(C)C(C3C(C)(C)C3(C)C)=O)C2)ccc2c(n1)NCC2 C1(C(=O)NCCOCC(=O)OC)CCCC(NC(C2CC2(C)C(F)F)=O)C1 N1(C(C2(CC#C)CCOCC2)=O)CCCC(O)(CCNC(=O)CC2=CCCC2)C1 N1(CC)CCC(NC(C2(NC(C3CCCC(=O)N3)=O)CCOCC2)=O)C(C)C1 C1(C(=O)NCCCN(c2cc(C)ncn2)C(C)(C)C)CC2CC(C)C2C1 CCC(CC(C)C)C(=O)NCC(C)(CNC(=O)C(n1cc(Cl)cn1)C)OC C=C(C)C1CCC(C)(O)C(N2CCN(C3CCOCC3)CC2)C1 c1(C(=O)NC(CNC(C2CCN(CC)CC2)=O)C(C)C)cc(C)c(C)c(F)c1 N1(C(=O)OC)CCC(C)(C(=O)N(C)CCNC(=O)Cc2cn(C)nn2)C1 N1(CCC2(OC)CCCC2)CCN(C(=O)NC2CC2(c2ccccc2)F)CC1 C1(CC(=O)N(C)CCOC2CN(c3ncc(F)cn3)C2)CC(=O)NC(=O)C1 c1(C(=O)NC2(C)CC(NC(C34CC(C)C3C4)=O)C2)nc(C2CC2)n2ccncc12 C(C(=O)NCC=CC)(N(C)C)C1CC1.C1(NC(=O)C=CC(C)(C)C)(CO)CCC1 C(CN=C(NCC(F)(F)CO)NC1CCCS(=O)(=O)C1)C1CCS(=O)(=O)C1 C1(NC(C(F)=CC)=O)CCCC1NC(c1ccc(CC)[nH]1)=O C(=O)(CC(C)(C)N(C)C(c1cnc(CC)o1)=O)NCc1onc(CC)n1 Cc1cc(CN2CC3C(C(N4CCC(F)CC4)=O)C3C2)cc(C)n1 S(=O)(=O)(c1ccc(N)cc1Cl)NCC1OCC(C)C1.C1(N(C)C)(CO)CCCC1 c1(-c2cc(C(=O)NCC(Cn3cc(C4CCOC4)nn3)OC)sn2)ccc(Br)cc1 C(C(C)(O)CCNC(=O)CN(C(=O)C(C)N=[N+]=[N-])C(C)C)OC c1(C(=O)NCC2CC(NC(c3cc(C)sc3)=O)C2(C)C)ccc(F)c2ccsc12 C1(NC(N)=O)CCOC(NC(CNC(C2C(C)(C)C2C(=O)NCCO)=O)=O)C1 c1(C(N2CCN(C3CN(C(c4c(C)con4)=O)C3)CC2)=O)ccc2nccnc2n1 C1(C)(C(N2CCC(OC(C)C)CC2)=O)CN(C(=O)CC2(C)CCOC2)C(C)(C)C1 C(C)(CO)(C(=O)NC1C(C)CCC1C)NC(Cn1c(C)nnn1)=O Cc1c(C(N2CCN(C)C(CNC(C3CCCCC3)=O)C2)=O)sc(Cl)c1Cl C(=O)(C1=NOC(C)C1)N1CC(OC(CNC(c2ccc(CC(C)C)nc2)=O)(CC)CO)C1 c1(CC)nc(=N)[nH]cc1C(N1CC(OCC(=O)NC2CN(C(C)=O)CC2C)C1)=O C1(NC(C(C)(C)SC)=O)CCC2(CCCN(C(c3c(C)ccc(Cl)c3N)=O)C2)C1 S(=O)(=O)(c1ccccc1OC(F)(F)F)NC(COC)CO C(=O)(C1=C(C)CCOC1)NCC=CC(N1CCCC(CCCC)C1)=O C1(NC(CC(C)OC)=O)CN(C(=O)Cc2ccc(C(N)=O)cc2)CC1OC Cc1c(C(N2CCC(N(C)C(C3CSCCS3)=O)C2)=O)cncc1Cl N1(Cc2ccc(OC)nn2)CC2CCN(C(c3ccc(C)cc3C)=O)C2C1 Cc1ccc(N)cc1C(=O)NCc1csc(CNC(=O)C(C)(C)F)n1 C1(CNC(C(CSC)OC)=O)(NC(c2cc(=O)cc[nH]2)=O)CCCCC1 c1(C(=O)NC(C2N(C(C(C(=O)NC)(C)C)=O)CCC2)(C)C)ccc(F)c(F)c1F c1(NC(C2CC3C=CC2C3)=O)nccc(C(N)=O)c1[N+](=O)[O-].CC1CN1 c1(C(N2C(c3cn(CC(C)O)nn3)CCC2)=O)c[nH]c2nc(Br)ccc12 C(C)(N=c1nc(N2CCSC(C)C2)c2sccc2[nH]1)c1c(COC)cccc1 CCC(C(=O)N(C(C)CNC(c1cocn1)=O)C)C1CCOCC1 Nc1sc(C(=O)NC2CCCCC2NC(=O)CSC2CC2)nc1-c1ccccc1 Cc1nc(C(=O)NC2CC(NC(c3csc(C(C)N(C)C)n3)=O)C2)c2ccnc-2[nH]1 Cc1cc(=NC2CC3CN(C(c4coc(S(N)(=O)=O)c4)=O)CC23)[nH]c(Cl)n1 CC1(NC(C2CC2c2ccncc2)=O)CCN(C(C2(C)CC2(F)Cl)=O)CC1 CN(S(=O)(=O)N1CCCC(C(F)(F)F)C1)CCC1CCOC1 N1(C(CC2CC(=O)CCC2)=O)CC2CC(NC(=O)CCC3CCC(=O)N3)CC2C1 N1(C(C(C)OCC=C)=O)CC2(CCC(NC(c3ccc(OC)c(F)c3)=O)CC2)C1 C(C1CN(C(=O)C(C)CC(F)F)Cc2ccccc21)NC(CC(CCC)O)=O c1(C(N2CCC(COC)(NC(=O)CC3CCCO3)C2)=O)ccc(F)c(C(F)F)c1 C(C)(CN=c1[nH]c2c(F)cccc2o1)NC(c1ccc(CC)c(C)c1)=O N1(OC(c2ccc(CN(CC=C)C)cc2)=O)CC(=O)CC(C)C1 C(=O)(C(F)CC(C)CC)N(CCN(C(CCOCC#C)=O)C)C c1(CC(N2C(Cc3cn(CC)nn3)CCC2)=O)cccc(NC(CCCC)=O)c1 C1(CC)COCCN1C(=O)CC1CCCCC1NC(C1(SC)CC1)=O C1(C(C(=O)NCC(=C)C)N(CCCO)C)CC2CCC1O2 CC(C)CC(O)CC(=O)NC1CCC1C(=O)NCCC(=O)NO Cc1cc(C(=O)NC23CCN(C(C4CC5C(C4)C5(F)F)=O)CC2C3)cc(Cl)c1 n1(CC(=O)NCC(CC)N(C)C(c2cc(C)n(CC)n2)=O)nc(C)n(C)c1=O C=CC(C)CC(=O)N1CCCC(C(C)(C)C(=O)NC2CC=CCC2)C1 C#CCC(C(=O)OCCCc1ccc(F)cc1)NC(=O)CCC(C)=O c1(C(=O)OC)cc(N2CC(O)(C(C)NC(=O)C(c3ccccc3)C)C2)nc(C)n1 n1(C(C)C)ncc(F)c1C(=O)NCC(CO)NC(=O)C(Cc1ccccc1)N(C)C c1(OC)ncnc(OC)c1C(=O)NCC12CCC1CN(C(C1CCO1)=O)C2 c1(C(=O)NC2CC(NC(c3nc(C#C)sc3)=O)C2)cc2cc(C)c(C)cc2o1 C=C(C)C(N)C(=O)NC(c1ccc(C)cc1)c1nc[nH]n1 CCS(=O)(=O)CC(=O)NC(CNC(=O)Cc1nn(C)cc1Cl)CO C1(NC(C(c2ccc(O)cc2)C)=O)CCCN(C(=O)Cc2ccnc(O)c2)CC1 Cc1ccc(Cl)c(NC(N(C)C(C2CCOC(C(C)(C)C)C2)=O)=O)c1 C(=O)(C(CN(C)C)C(C)C)NC(CN1CCC(NC(CCC(=C)Cl)=O)CC1)C CCC(O)C(C)C(=O)NCc1ccc(C(N2CC(c3ccc(C)cn3)C2)=O)o1 C1(C(=O)NCCN(C(c2c(C)noc2C(C)C)=O)C)CCc2nncn2C1 c1(C(N2CCN(c3ncc(C)cn3)C(C(C)C)C2)=O)cc(Cl)cc(Br)c1Cl C1(NC(C(c2c(C)noc2C)C)=O)CC2(CCN(C(C3CC3C#N)=O)C2)C1 CC(CCC(=O)N1CCCC1)C1CCC1NC(=O)C(C1CCOCC1)F C1(C(=O)NC(CNC(c2cnc(OC)s2)=O)C)(N(C)C)CCCSC1 C1(C(N(C(CNC(c2[nH]ccc2Br)=O)C2CC2)C)=O)CCCCN1C CCC(C(=O)NCCC1CCCN1c1nnc(C2CCCC2)s1)SC C1(C(N(C2CCCN(C(=O)CC=C(Cl)Cl)C2)CC)=O)CCC2CC1CO2 C1(CCCNC(c2n(CC)nnc2)=O)CN(C(=O)CC23CCCC2C3)CCO1 C1(NC(c2cc(CC(C)C)on2)=O)CCN(C(=O)COCC(F)(F)F)C1C C(CNC(C1CCC(=O)NC1)=O)(C(C)(C)C)NC(C1(CCC)CC1)=O C1(CNC(CCC(=C)Cl)=O)CCN(C(c2cc(C(C)=O)c[nH]2)=O)CC1(F)F C1(CC)(CC)CC(NC(=O)Cn2cnnc2)CN1C(=O)CNC(=O)Cn1cncn1 C(C)(C(=O)N1CC(c2noc(=O)n2C)C1)(C(C)C)NC(=O)OC(C)(C)C C1(C(=O)NCC2(C(=O)NCc3ccccc3)CC2)CCCOCC1 N1(C(Cc2c(C)ccs2)=O)CC(C2(NC(=O)C(C)NC(C3CCCC3)=O)CC2)C1 c1(C(=O)OCC)cncc(C(N2CC(N(C)C)C2)=O)c1.C(=O)(C(CO)N)OCC C(=O)(C#CC1CCOCC1)N1CC(C)(OCC(=O)NCCC(COC)O)C1 c1(C(=O)NC2CCCN(C(CC3N(CC)CCC3)=O)C2C)cc2n(n1)CCNC2=O Cn1nccc(C(N2CCCC2c2cn(Cc3ccno3)nn2)=O)c1=O c1(C(=O)NCCC2(O)CN(C(c3n(CC)ncc3Cl)=O)C2)c(C)ccc(C)c1O C(=O)(C(CCc1ccsc1)N1CCCC(CN(C)C)C1)NCCCC CC1=C(C)CC(C(=O)N(C)CC2COCCN2C(c2cc(F)ccc2Cl)=O)CC1 Cc1ccc(CC(N2CCC(N(C(=O)C(C3CCCCC3)F)C)C2)=O)cc1O c1(C(=O)NCCC2C(C)CCCN2C(=O)CN(C)C)cnc2ccccc2n1 C(=O)(C(CO)C(C)(C)C)NCCC1CCN(C(C(CC(C)C)NC(C)=O)=O)C1 c1(C(N2CCC(C)(C)C(NC(c3cnc(O)o3)=O)C2)=O)ccc2cccnc2c1 c1(NC(C2(C)CN(Cc3ccc(F)c(Br)c3)C2)=O)cccn2ccnc12 C=CC1CN(C(=O)C(CC2CCOCC2)NC(=O)CC2COCCO2)CCO1 CCCC(C)(C)C(=O)N1CCC1C(N1CCOC(C(C)C)C1)=O Clc1nc(-c2ccc3c(c2)CCNC3)cc2occc12 CC(C)CC(CNC(C1CCC(N(C)C)CC1)=O)NC(c1ccc(CF)cc1)=O C(CCCC(C)NC(c1c[nH]c(=O)cn1)=O)NC(C(CC)N(C)C)=O c1(NC(CCC2(C)N(C(c3ccn(C)n3)=O)CCC2)=O)cccc(F)c1F C(CCC)(C(=O)N(CCNC(=O)C(c1cccc(F)c1)O)CC1CC1)=CCC n1(CC)c(C(N2CC(C)(C(=O)NC3(c4cccs4)CC3)C2)=O)cnc1O C1(NC(c2ccc(=O)n(O)c2)=O)CCCCN(C(C2CN3CCC2CC3)=O)C1 c1(C2C(CNC(=O)NC(c3ccccc3)C3COC3)C2)ccccc1 c1(C(N2CCCC(NC(CC3CC(=C)C3)=O)C2C)=O)nc2ccccc2n1CC c1(C(N2CC(NC(C3ON=C(CC)C3)=O)C(F)C2)=O)cc2ccccc2[nH]1 C1(NC(c2c(OCC)cccc2)=O)CC2CN(C(=O)Cn3ccc(C)n3)CC2C1 N1(C(C(COCC)C)=O)CC(C2(NC(=O)CN(C)S(N)(=O)=O)CC2)C1 C(C(COC)C(=O)NCC1(CCCNC(=O)Cc2cnc(C)s2)CCCC1)OC C(=O)(C(C(C)(C)C)NC(N)=O)NC(CC(C)NC(C1CCOC1)=O)C c1(-c2cn(CC3CCN(C(c4ccoc4I)=O)C3)nn2)cc2cccnn2c1 C=C(C)CC(C)C(=O)NCCN(CCC)C(c1ccc(OC)cn1)=O N1(C(c2c(CC)cco2)=O)CCN(C(=O)C=CC(C)CC)C2CC12 c1(OC)ncc(Br)c(=NCC2CCC(NC(c3ccccc3CO)=O)C2)[nH]1 c1(OC)cc(C(N2CCC(C)(CNC(C3CCNC3=O)=O)C2)=O)cc(F)c1 C1(NC(CCC#C)=O)CC2CCC1N2C(=O)CCc1ncc(C)[nH]1 C(=O)(C(CC(C)(C)C)NC(C1CC1OC(C)(C)C)=O)N1C(CC(=O)NC)CC1 N#Cc1sccc1C(=O)NC1CCC(CC(=O)Nc2ncccc2F)C1 CCC(C)(C)C(=O)C(=O)NC(CC1CC1)C(=O)NC(C1CCCC1)CO C(=O)(C1=CCCOC1)NC(C(=O)NCC(C1CCCCC1)O)C1CC1 C1(NC(C)=O)CN(C(=O)COCC2CC2)CC2(CCC2)C1 C=CCC(C(=O)OCC)NC(=O)CC1CCCC(NC(=O)C=CC(=O)N(C)C)C1 C1(N(C(=O)C(=O)Nc2cc(F)ncc2Br)C(C)C)CC(C)OC(C)C1 CN1CCC(NC(=O)C(F)C2CC(NC(c3ccn(C4CC4)n3)=O)C2)C1 Cc1cc(Cl)nc(N)c1C(=O)NCc1ccc(C(C)NC(C2CCCS2)=O)cc1 C(=O)(C(C)(O)CC(C)C)NC1CN(C(c2c(-n3c(C)nc(C)n3)cccc2)=O)C1 C(CC(CC)C(=O)NC(CCNC(C1CC(F)C1)=O)C(C)C)=CC C1(NC(c2c(C(C)C)ccs2)=O)CC2CC(NC(=O)C(C)c3ccsc3)C2C1 C(CCC1CC1)(C(=O)NC1(CC2CCC2)CC1)NC(c1cc(COC)[nH]n1)=O N1(C(c2cn(CCC)nn2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CC(C)C1 C(=O)(C(C)CCCCOC)N(C(CC)C(C)C)C(C)CNC C1(C(=O)NCC(CNC(c2c(CC)occ2)=O)O)Cc2nncn2C1 C(CC(C)C)(C(=O)N1CCC1C1CCOCC1)N(C(c1[nH]cc(C)c1)=O)C N1(C(C2(NC(=O)Cc3csnn3)C(C)(C)C2)=O)CCC(C2CCCC2)C1 C12(C(N3CCC(CCOC)CC3)=O)CCN(C(=O)C(F)=C(C)C)CCC1C2 CC(CN=c1[nH]c(=NCC2CC2(C)C)[nH]c2c1COCC2)Oc1ccccc1F C1(NC(C=CC(=O)OC)=O)CN(C(=O)C(c2ccccc2)NC(N)=O)C(C)(C)C1 C1(CNC(c2n[nH]c3c2CCC3(F)F)=O)CC2CCCCC2N1C1CC1 C1(NC(CCCN(C)C)=O)CN(C(c2scnc2C(C)(C)C)=O)CC1(C)C C1(C2CCCOC2)(NC(=O)Nc2ccc(F)cc2Cl)CC1 n1(CC)nc(C(=O)NCC2CC2CNC(C2(C)CCOC2)=O)c2ccccc12 C1(NC(CCCOCC)=O)CCCCN(c2cnc(OCC3CC3)cn2)C1 C1(CNC(=O)CSc2nc[nH]n2)CCCCC1C(=O)NCCCCn1ccnn1 C1(CNC(CCC#C)=O)C(O)C(O)CN1C(=O)CSCc1ccccn1 CCCCCC(=O)N1CCC(C(C)NC(=O)CS(=O)(=O)NC2CC2)C1 C1(C#N)(C(=O)NCCOCCCNC(c2nc(CCC)sc2)=O)CC12CCC2 C=C(C)CC(C(=O)NCc1ccn(C)c(=O)c1)NC(=O)C(C)NC=O CCC(CCC(=O)NC(c1nncn1C)C)NC(=O)Cc1ccccc1F CCC(C(=O)NC1CN(C(c2ccc(OC)nc2F)=O)CCC1CO)C(C)C c1(C(N2CCC(C3CCCN3C(=O)CCn3ccnc3)C2)=O)ccc(O)nn1 C(=O)(C(C)C(C)(F)F)NC(CC)(C)CNC(c1sc(C2CCCC2)nc1C)=O c1(OC)cccc(SCC(N2CCC(C)(NC(=O)CCNCC(F)(F)F)C2)=O)c1 C1(NCC)CCC(N=c2[nH]c3c(c(=NCc4cscc4C)[nH]2)COC3)C1 N1(C(C)=O)CCCCC1C(=O)NCC1CC(NC(=O)C(C)C(F)F)CO1 C1(OS(CC(C2CCCC2)OC)(=O)=O)CCCCCCC1 C1(NC(C(CC)SC)=O)(CC)CCN(C(=O)Cc2ccccc2OC)CC1 c1(NS(CCN(C(C)C)Cc2ccccc2F)(=O)=O)c(Cl)nc(Cl)n1C S(=O)(=O)(c1ccccc1[N+](=O)[O-])NCC(N1CC(CNC(C=CSC)=O)C2C1C2)=O c1(SC(C(=O)OCC)CC)nc(O)c2cnn(C(C)(C)C)c2n1 c1(CN2C(C(=O)OC)CSC2C(F)(F)F)ccc2c(O)nccc2c1 c1(C(N2C(CNC(C(COC)NC(C)=O)=O)C=CC2)=O)cnc2n1CCOC2 c1(C(=O)NCCCOCCNC(=O)C=Cc2cnc[nH]2)sc2cccnc2c1Cl N12CCC(CO)(CC1)NC(=O)c1scnc1CCC2=O.C1(NC(C)=O)CC(C)(C)C1 C1(COC)(NC(c2cnn(C(C)C)n2)=O)CCCN(C(c2cnccc2C)=O)C1 C1(CNC(=O)NC2CCCC(CN3CCOCC3)CC2)CCC2(CC2)CO1 c1(OC)ncc(NC(C2(C)CCN2C(c2nccc(C)n2)=O)=O)cc1Br c1(Sc2cccc(C3(OC)CC3)c2)ccc(Cl)cc1Cl.C12CCN(C1)C(=O)N2 C(=O)(CCCCC#N)N1CCC(CCC(=O)N(CC(=O)NC(C)(C)C)C)CC1 c1(OC)cc(C(=O)NCC2C=CCN2C(c2cnc(Cl)[nH]2)=O)cc(Cl)n1 C1(C(=O)N2C3CC2C3)CCOC1CC(=O)NC1CC1.C1(C(N)=O)(SC)CCC1.C(F)F c1(C(=O)NC2CC3CC(NC(COCC#C)=O)C3C2)noc2cc(F)ccc12 CCC(CC)CC(=O)NC1CCC1NC(C1(c2cccs2)CC1(F)F)=O CC1CC(NC(C2NC(=O)OC2(C)C)=O)CCN1C(=O)CN1C(=O)CN(C)C1=O C(=O)(C1CCc2nccn21)NC(c1ccc(N(C)C(=O)Nc2cnn(C)c2)cc1)=O c1(C(=O)NCC2(C(=O)NC(C#N)C(N)=O)CC2)cc(Cl)sc1Cl Cc1cc(O)ccc1C(=O)NC1CC1NC(=O)C(C)Cn1ccnc1 c1(C(N(CCNC(=O)CCC2CCC(C)O2)CC)=O)c2c(c[nH]c1=N)CCC2 C=CCC(C(=O)NC1(C(=O)N(C(C(N)=O)C2CC2)C)CC(O)C1)C(C)C Cc1ccc(Cl)cc1C(C(=O)NCCC#N)N(C(C#N)CC)CC#N C1(NC(c2cc(CF)on2)=O)CCC2(CCN(C(=O)C3=CCCOC3)CC2)C1 C1(N(C(Cc2ncc(C)s2)=O)C)CCCN(C(c2cnoc2C)=O)C1 CC(F)CC(=O)N(C)CC1CCN(C(=O)C(n2cc(Cl)cn2)C)C1 Cc1cc(C#N)sc1C(=O)NC1CCN(C(c2ccn(CC(C)C)n2)=O)C1C c1(C(=O)NCCNC(C2CC3C=CC2C32CC2)=O)ccc2n[nH]cc2c1 C(=O)(CCCC(C)NC(c1ncn2c1CCC2)=O)N(C(C)CC1CC1)C C1(OC)CC(CNC(c2csc(=N)[nH]2)=O)N(C(=O)C(C)C2CC2)C1 c1(OCC)cc(OC)cc(N2CCC(NCc3cc(C(F)(F)F)ccc3F)C2)c1 C=C(Br)CC(C)(C)C(=O)NC1CN(C(c2cnn(C)n2)=O)CC1CO c1(CC(=O)NCCCC2CCCN2C(C2CCSC2)=O)sc(O)nc1O C(=O)(C1=C(C)CCOC1)NC(COCC)C(=O)Nc1cc(C)cnc1C c1(-c2cccc(OC)n2)ccc2c(C(=O)Nc3cnnn3C)nn(C)c2c1 Cc1ccc(C(O)C(=O)OCCC2CCCOC2)cc1 c1(C(=O)NCc2ccc(CN(C(CC=C)=O)C)cc2)noc2c1COCC2 Nc1cc(F)c(C(=O)NCC2(CCNC(c3cc([N+](=O)[O-])n[nH]3)=O)CC2)c(F)c1 CN1N=C(C(=O)N2CCN(C(c3ccc(I)cc3Cl)=O)CC23CCC3)CCC1=O c1(-c2onc(C(C)C(N)=O)n2)cnccc1C#N N1(C(c2ccc(-c3ccc(CC)cc3)o2)=O)CCN(c2nnc(C)o2)CC(O)C1 N1(C(C2ON=C(C)C2)=O)CCC(C2CN(C(=O)CN3CCCCC3)C2)CC1 Cc1cccc(C)c1CCOC(=O)CCCN1CC(c2ccc(Cl)cc2)C1 c1(CNC2CN(C3CN(C(c4cccs4)=O)C3)C(=O)C2)c[nH]c2cccnc12 C(CCCCCC(=O)NCCc1csnn1)NC(C(N1CC(C)C1)C)=O C12(CNC(C=C(C)C(F)F)=O)CCC1CCN2C(c1n[nH]c(=N)s1)=O C12(CNC(c3nc(C(C)(C)C)[nH]n3)=O)CCCC1CCN2C(C1CCCC1)=O N1(C(COCC=C)=O)CCC2(CC1)C(C)C(C)OC2=O.C(C)(CC)NC(C)=O N1(C(c2cc(C(=O)OC)on2)=O)CCCCC(NC(=O)Cc2c(C)n[nH]c2C)C1 N1(C(C2N(C(CC3(OC)CCC3)=O)CCCC2)=O)Cc2ccc(Cl)cc2C(C)C1 C1(C(=O)NC2CC(CNC(=O)CCc3cccnc3F)C2)CCC2(CCC2)O1 C1(C)(CC(=O)N(CCCNC(=O)CC(F)(F)F)C)CCS(=O)(=O)N1 N1(C(c2ccc(C(=O)OC)s2)=O)CCC(N(C)C(c2cc(C)co2)=O)C(C)C1 N1(C(CCOC)C)CCn2c(C(F)F)nnc2C1 c1(CC(=O)NCC(CC)(C)NC(=O)C(c2cccc(O)c2)C)ccccc1OC C=CC(C)C(C)C(=O)NCC1(CO)CCN(C(C2(C3CCC3)CC2)=O)CC1 c1(C(=O)NCC2C=CC(NC(=O)CC34CCCC3C4)C2)cc2ccncc2c(O)n1 c1(CNC(C2C(OC(C)=O)C2)=O)cc(C(=O)NCC(C)(O)CO)cs1 C1(C(N(C)Cc2ccc(F)cc2)=O)C(C2CC2)CCN1C(=O)CCc1ccoc1 N1(C(c2cc(CO)[nH]n2)=O)CCC2CCCC12C(=O)NCC1CCC1(F)F N1(C(CCC2CCC(C)O2)=O)CCCC(C2CN(C(C3OCCC3(C)C)=O)C2)C1 C1(NC(C2CCC(=O)NC2)=O)(CNC(=O)C(C2CC(F)(F)C2)O)CCCCCC1 N1(C(C2CN(C(CCC(=C)Cl)=O)CC2(F)F)=O)CCC2CC1C(=O)O2 C1(NC(C2CCN(CC)CC2)=O)CC2CCC1N2C(c1cnn(C(C)(C)C)c1)=O c1(-n2cc(C3N(C(CC4CCC(OC)CC4)=O)CCC3)nn2)cccc(F)c1F O=C1CCC(C(=O)NC2CCC2C(=O)NCCN(CCO)CCO)CCO1 C1(NC(c2ccc(N(C)C)nc2)=O)(CNC(C2(O)CCSC2)=O)CC2CCC1C2 C=C1CCC(C(=O)N(C)CC=CC(=O)NC(CO)C2CCC2)CC1 CCC(CN(C)C)CC(=O)N1CC(O)CC1CNC(=O)CCn1ccc(C)n1 c1(CC)cc(C(N2CC(NC(c3ccc(OC(F)(F)F)nc3)=O)C2)=O)ccc1Cl C(=O)(CC(C1CC1)NC(C1CC(C)N1C(=O)C(C)(C1(C)CC1)OC)=O)NCC C(C(C(=O)Nc1cn(C)nc1C1CC1)C(C)(C)C)NC(C(CC=C)C)=O N1(C(COC(CC)C)=O)CCN(C(=O)COC2CCC2)CC1CCO C(=O)(CC(C(F)F)n1ccnc1)N1C(C(N(C(C)C)C)=O)CCC1C C(=O)(CCCC(F)(F)F)NC1(C)C(C(N(C)CC2(O)CCC2)=O)CCCC1 C1(C(=O)NCC2CCN2C(=O)COc2ccccc2)(OC)CCCCCC1 c1(CCC(=O)N(C2C(C)CCNCC2)c2ccncn2)ccc2ccn(C)c2c1 C(=O)(CCC(CC)NC(c1cccnc1)=O)N(CCCC)CC C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCC1CCN(C(CC2(C)CCOC2)=O)CC1 N1(C(CCCCC#C)=O)CC2CC(C)N(C(=O)Cc3cc(CC)nn3C)C2C1 C12(NC(CCN(C)CCO)=O)CCCN(C(C3(CC4CC4)CCC3)=O)CC1C2 CC1(C)C2CCC1(C)CN(Cc1n(Cc3ccccc3OC(F)(F)F)ccn1)C2 N1(C(C2(C(C)(F)F)CCC2)=O)CC(NC(C2CCC3(CCC3)CC2)=O)CC(O)C1 N1(C(C=CC=CCC)=O)CCC2CCN(C(=O)Cc3c[nH]ccc3=O)CC2C1 C(=O)(C1=CCCSC1)N(C)CC1CCN(C(C(CC)NC(N)=O)=O)CC1 c1(C2C3N(CCC3)C(=O)N2)ccccn1.C1(CO)CC(CCn2cccn2)C1 O=C(O)CC(O)C(=O)N1CCOC(c2cccc(C(F)(F)F)c2)C1 N1(C(CCCOC(C)=O)=O)CCCC(CCNC(C2CCCC3(CC3)C2)=O)CC1 C#Cc1cc(C(N2CCC(NC(C3CCCN3C3CC3)=O)C2)=O)cc(Br)c1 Cc1ccnc(C)c1NC(C1CCCCN1C(=O)CCc1cnoc1)=O C(=O)(C(CC(=O)NCC(O)CC(F)(F)F)NC(=O)OC)OCC(C)(C)C N1(C(C2C(CCC)CCC2)=O)CC(NC(=O)CCc2cnc[nH]2)C2CCCC2C1 c1(OC)cccc(C(=O)N(C)CCOCCCN(C)C(C2CC3CCC2C3)=O)n1 c1(NC(CCC)C)ncccc1S(=O)(=O)NCC(CO)C1CCC1 N1(C(C(=O)NCC)=O)CC2CC1CCC2NC(C12CCCCC(OC)(C1)C2)=O c1(CC(=O)N(CC(CC)NC(=O)COC(C)(C)CC)C)ccc2c(c1)CCCO2 C1(CC(=O)NCC(CC(C)C)NC(C(=O)NCC)=O)CC(=O)c2ccccc2C1 Cc1cc(Cl)c(Cl)cc1C(N1CCC(O)(C(=O)Nc2cnnn2C)C1)=O N1(C(C(CC=C)Cc2ccccc2)=O)CC(NC(=O)C2=CCC2)C(S(C)(=O)=O)C1 C1(C(=O)NC2CC(NC(c3cccc4cc[nH]c34)=O)C2)CC2CCC(C1)S2(=O)=O c1(C(=O)NC(C(=O)N2C(CC(C)C)CC2)Cc2ccco2)cncc(Cl)c1 Nc1ccc(C(=O)NCC(C2CC2)NC(c2coc(Cl)n2)=O)c([N+](=O)[O-])c1 c1(C(N2CCC3CN(C(CC4(C)CC4)=O)C3C2)=O)cccc2c(Br)ccnc12 Cc1cc2ccccc2n1CC(N1CCC(CO)=C(F)C1)=O.C1CS1 c1(CN2CCCC(C(=O)Nc3ccc(CC)cc3)C2)cc(Cl)c(O)cc1O CCCC(CC)C(=O)N1CCC(F)(F)C1c1ccc(NC(=O)CSC)cc1 CC(=NO)c1sc(NC(c2ccccc2CC#N)=O)nc1C N1(C(CCC(C)NC(=O)Cn2ncnn2)=O)C2CCCC1COC2 c1(C(=O)NC(C)C(CO)NC(=O)C(O)C(C)(C)C)cccc2c1CCC2 N1(C(CC(CC(=O)OC)C)=O)CCC2OCCN(C(=O)C=CC3CCCC3)C2C1 c1(CCNCC(COC)O)cccc(NC(=O)OC(C)(C)C)n1 c1(C(=O)NCCN(C(c2c(CC)ocn2)=O)CC)cnn2c1OCC2 C1(NC(CC=C(C)C)=O)CCCN(C(=O)CC2CCC(C3CC3)O2)C1 C(CNC(c1ccccn1)=O)(CC(F)(F)F)NC(c1cc(Cl)nc(Cl)c1)=O c1(N(C(C)C(F)(F)F)CC)nc(C)cc(C#N)n1 C1(NC(C(C)(C)N(C)C)=O)CCN(c2ncnc3c2COC3)CC(C)(C)C1 N1(C(C(C)OCC#C)=O)CCN(C(c2c(C)[nH][nH]c2=N)=O)CC1C(F)F c1(C(N(C)CC2CCN(C(C(CC)O)=O)C2)=O)cncc(F)c1C c1(CNC(=O)Nc2ccc(C3CCC3)cc2)cc(F)c(F)cc1Cl Cc1cc(C)c(C(=O)NC2(C3CCCN3C(=O)CC3COC(=O)C3)CC2)o1 N#Cc1nc[nH]c1C(=O)NCc1ccc(Cn2cc(C3CCCO3)nn2)cc1 c1(C(=O)NC2CC3(C(NC(=O)CC45CCCC4C5)C3)C2)cccc2nccnc12 C1(C(=O)NCC2CCN(C(CCOCCOCC)=O)C2)CCCC(=O)O1 c1(NC2(CNC(c3cccs3)=O)CC2)ncnc2c1CCC2 C1(C(=O)Nc2ccc(OC)cc2C)CCC2(CN(c3ncnc4sccc34)C2)O1 CON1CCC(C(N2CCCC(C)(NC(=O)Cc3ccc(F)cn3)C2)=O)CC1 CC#CCC(C(=O)NOCCCO)NC(=O)CC(CCC(C)C)NC N1(C(c2ccc(SCC)cc2C)=O)CCC2(CCCC2NC(=O)CCC2CC2)C1 C(C)(CS(=O)CC)N(CC(C)NC(c1cnc(C(C)C)[nH]1)=O)C C(=O)(CCCC(C)C)N1C(C2(C(=O)NCC3(C)N=C(C)SC3)CC2)CCC1 C1(N(C(c2cc(CC)[nH]n2)=O)C)CCN(C(=O)CNC(=O)OC)CC1C Cc1csc2ccc(C(N3CC(CO)(NC(C4C(C)OC(C)C4C)=O)C3)=O)cc12 Fc1cccc(CNN2CCN(c3ccccc3)C(CC3CCCCC3)C2)c1C C(CC(C(=O)N1CCN(CC)CC1)NC(C1(CC)CC(OC)C1)=O)OCC N12CC(C3(CC3)C1)C2=O.Cc1ccnnc1NC(=O)COc1ccccc1 C1(NC(Cc2c(C)non2)=O)CCC(N(C)C(C2CCC(F)C2)=O)CC1 Cc1ccccc1C=CC(=O)NC1CCCCN(C(C2CS(=O)(=O)C2)=O)C1 c1(C(=O)OCC)nc(N2CC3C(NCc4cccnc4)C3C2)cc(Cl)n1 c1(SC)cc(C)c(C(N2CCCC2C2CCCOC2)=O)s1 c1(C(=O)NCCCN(C(C(C)SCC)=O)C(C)C)cc2ccc(F)cc2nc1C C(CCCCC(=O)NN1CCCOC1=O)n1cc(C(C)(C)C(=O)O)nn1 C#Cc1ccnc(C(=O)NC2CCCN(C(C3(OCC)CCOC3)=O)C2)c1 CC(CC(F)F)C(=O)N1CC2CC2(C(N2CCSCC2)=O)C1 C1(N(C(C2(C#C)CN(C(c3ccn(C)n3)=O)C2)=O)C)CCCCC1(C)C C(C(C)(C)C(=O)N1CC(O)(CCNC(=O)CNC(=O)CN(C)C)C1)SC N1(C(C(c2cnn(C)c2)C)=O)CC(NC(C2CC(n3cnnc3)C2)=O)CC(O)C1 c1(OC)cc(C=CC(N2CC(NC(c3ccno3)=O)CC2C)=O)ccc1O C1(NCC2CCN(S(C)(=O)=O)CC2)CCN(C(=O)COC2CC2(F)F)CC1F CC(CCNC(=O)C(C)CN(C)C)CCNC(c1cc(C2CC2)[nH]n1)=O c1(C(N2CCN(C(C(C=C)(C)O)=O)CC(CO)C2)=O)ccn2c(O)nnc2c1 N1(CCNC(=O)CN2CCN(C(=O)C(=O)NC3CC3)CC2)CCCNS1(=O)=O CC1(NC(C2CCN2C(=O)C(O)C2CCC2)=O)CC=CCC1 c1(-n2ccc(C(=O)NC(CCCC)CNC(=O)CC(F)F)n2)c(C)nn(C)c1C CC(CC(=O)NCC1(CC(=O)NOCC(N)=O)CC1)C(F)(F)F C(=O)(C1=CC2CC(C1)CC2O)N1CC(OCCNC(=O)Cc2n[nH]c(O)n2)C1 C1(NC(C(SC)SC)=O)CC2CC1CN2C(=O)CCc1cn(C)cn1 c1(C(=O)NC23CC(CNC(C(CC#C)O)=O)(OC2)C3)c[nH]c2ccccc2c1=O C(=O)(C(CC(C)(C)C)OC)NCC(CCNC(C(CCC)NC(C)=O)=O)OC Cc1c(NC(=O)C(C2CCCO2)NC(C2CCC(=O)NC2)=O)cnn1C1CC1 C(=O)(CC(C)N(C)C(c1cc(C)ns1)=O)N(C1CC(OCC)C1)C Cc1cc(=NCC(C)(C)n2cccn2)[nH]cc1S(=O)(=O)NCCN(C)C.C1CN1 CCCC(C)C(=O)N1CCC1C(=O)NCC(O)COCC N1(C(C(C)OC2CCCCC2)=O)CC(NC(c2cccc(Br)c2)=O)CCC1C CC1CC(NC(c2ccc(CO)s2)=O)CCN1C(=O)CCC1CCCO1 c1(C(=O)NC2C(NC(C(c3cccc(Br)c3)C)=O)CCC2)cc2n(c1)CCC2 C1(CNC(C2(C)CCN(C(C(C=C)OC)=O)C2)=O)CC(=O)N(C)C1=O CCC(C)(COC)C(=O)N1CCCC1CNC(=O)Cc1cccc(C(C)C)c1 N1(C(C2CC3(CC(NC(Cc4ccc(C)o4)=O)C3)C2)=O)CC2OCCN(C)C2C1 C1(NC(=O)C(F)C2CCCC2)CC12CCN(C(c1csc(O)n1)=O)CC2 C1(C(=O)NCCOCCC(C)C)CCC(C2CC2)N1C(=O)Cc1ccoc1 c1(OC)noc(C2CC2)c1C(=O)N(C)CC1COCCN1C(=O)C1CC1 C1(CNC(C(CC)SC)=O)C(C)CCCN1C(=O)CC1CCC(C)C1 c1(-n2cc(CN(C(Cc3c(C)nsc3N)=O)CC)nn2)ccc2occc(=O)c2c1 N1(C(C2CN(C(C)C)C2)=O)CCN(C(C2C3CC3C3CC23)=O)CC1C c1(C(C(=O)NC(C)C(CO)NC(=O)C(F)C(F)(F)F)=O)cc(F)c(F)cc1F CC(C(C)(C)NC(c1ccc(CN2CCCC2)o1)=O)NC(=O)COc1ccsn1 C1(NC(=O)NC(C2CCCCO2)C2CC2)CCOCC12CCCC2 C1(NC(C(C)CC(F)F)=O)CCC2(CC1)CN(C(C1CCCCC1)=O)CCO2 c1(CC)cc(C(=O)NCCN2CCC(NC(C3(C)CCCC3O)=O)CC2)sc1C N1(C(C(C2CC2)OCC)=O)CCCC2(C1)CN(C(C1CCS(=O)(=O)C1)=O)C2 c1(CC)cc(C(N2CC3CC2(CNC(c2sc(C)cc2C)=O)C3)=O)nn1C C1(NC(=O)Cc2ccsn2)CN(C(=O)C2=CCOC2)C2(CCCOC2)C1 Cc1ccc(C)c(CNC2(CO)CCSCC2)c1 N1(C(C2C3N(C(CSCC=C)=O)C(CC3)C2)=O)CCc2sccc2C1 CCC(C)C(C)C(=O)N1CC2CC1CN2C(=O)CC1CCC(C)(C)CO1 N1(C(Cn2cccc(C)c2=O)=O)CCC2CC2(NC(=O)Cn2ccnc2C)CC1 N1(C(c2ccc(C)c(F)n2)=O)CCCN(C(C2(CO)CC2(F)F)=O)CC1C N1(C(C23N(C(C4C(C(=O)OC)C4)=O)CC(C2)C3)=O)CCC2(C=C(C(=O)NC)C2)C1 c1(C(N2CCC(NC(c3n(CC)ncc3)=O)C2)=O)cc(=O)n(C)cn1 n1(CCCOC)c(N2CCC(C3CCCO3)CC2)nnc1CCc1ccccc1 c1(C(=O)NCC2C(C)CN(C(C3COC(C)C3)=O)CC2)cc([N+](=O)[O-])cn1C CC(C)CC(O)C(=O)NCC1C2CN(C(=O)CCC(=O)N(C)C(C)C)CC12 N1(C(C2(CCC=C)CN(C(c3ccnc(C)c3)=O)C2)=O)CCC(CO)C(C)(C)C1 N1(C(Cc2cccc(C)c2)=O)CC(NC(C2CCCCN2C)=O)C2CCCCC12 c1(C(=O)NCc2c(CCNC(C(CCOC)C)=O)ocn2)c(C)nc(O)nc1C c1(C(=O)NCCCCCNC(CCCC(N)=O)=O)cnc2c([N+](=O)[O-])cnn2c1 N12CCCC3(C1)CN(C3)C(=O)C1(CC1)C2=O.CC1CCC(Oc2cnc(O)s2)CC1 C1(OC)CN(C(C2(CC3CC3)COC2)=O)CC1NC(=O)C=CCCc1ccccc1 C=CC(C)C(C)C(=O)NC1(CC=CC(=O)NCC2CC3(CCC3)CO2)CCC1 C1(O)(C(=O)NC(CCN(C(C2(SC)CC2)=O)C)c2cccs2)CCOCC1 C(=O)(CCCCC(N)=O)NCc1cn(C2CCN(C(CN(C)CCO)=O)C2)nn1 c1(C(=O)NCC(C)NC(C(CC)O)=O)cc2ccsc2[nH]1 c1(CC)noc(C(=O)N(CC(O)CN(C(=O)C(C)C2CCC2)C)C)c1C C1(NC(c2c(C)nn(CC)c2Cl)=O)CCCCN(C(=O)CC2CCOC2)CC1 c1(C(=O)NCCNC(CC2C(C)CCC2)=O)nnc(O)cc1O.C(c1ccnn1C)=C c1(CC2(NC(=O)N(C)SC)CC2(C)C)cc(Cl)ccc1Cl C(=O)(C(=O)CCC(C)C)NCC(CCC)C(=O)NC(C(C)(C)O)C1CC1 C(=O)(C1=COCCC1)N(CCNC(C1(C)CNC(=O)C1)=O)CCc1ccccc1 C(C(=O)N=S(C)(=O)c1ccc(C(C)C)cc1)N1CCC(NS(CCC)(=O)=O)CC1 C1(C(C(N2CCC(N(C(COC)C)C)C2)=O)C)CC2CCC1C2 C1(C(=O)NCC2CCCCN2C(c2n[nH]c(C(C)C)n2)=O)(COC)CC=CCC1 c1(C(=O)NC2CCN(C(c3c(C(C)C)ocn3)=O)C2)coc2c1C(=O)NCC2 C1(CNC(=O)CCN(C(C2CC(=C3CC3)C2)=O)C2CC2)CCCC(C(F)(F)F)C1 C1(C23CC(c4cn(NC(C5COCC5C5CC5)=O)nn4)(C2)C3)CC2(C1)CC(O)C2 C1(CC(=O)NCCN(C)C(c2ccccc2)=O)Cc2ccc(Cl)cc2C1=O N1(C(CC#N)=O)CC2CC2(CNC(=O)CCNC(c2ccc(O)cc2)=O)C1 c1(CC(=O)NCC#CCNC(=O)CC2CCOC2=O)ccc(F)cc1 C1(NC(=O)CC2CCC2)CN(C(C2CCCOC2)=O)C2(CCCC2)C1 C1(C(C)NC(c2nc(CC)sc2)=O)CN(C(=O)CCc2cscn2)CCO1 c1(C(N(CCn2cc(CCC3CCCOC3)nn2)CC)=O)nc(Br)n2ccsc12 Cc1ccc(NCC2CN(C(=O)NCC(=O)NC3CC3)C2)c(S(C)(=O)=O)c1 CC(CN1CCOCC1)C(=O)N1CCC(C(C)NC(C2CC(=C3CC3)C2)=O)C1 c1(C(N2CCC(NC(COC)=O)CC2C2CC2)=O)ccc2n[nH]c(C)c2c1Cl C=C(CNC(=O)C=CCNS(=O)(=O)CC)CCNC(=O)C(C)Oc1ccccc1 N1(C(CCOCCOCC)=O)CCC(N(C)C(C2CCC(C(C)(C)C)O2)=O)C1 CC1=CCSC1C(=O)NCC(C(=O)NC(C(N)=O)C1CC1)N(C)C Cc1[nH]c2ccnn2c(=O)c1CC(=O)NCC1(N(C(=O)C(C)(C)F)CC)CCC1 N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCCC(CN(C)C(c2cccs2)=O)C1 C(=O)(CCCCCCCCCO)NC1C2CC(CNC(C(=O)N(C)C)=O)(C2)OC1 c1(NC2C(NC(C(C)Oc3ccccn3)=O)CS(=O)(=O)C2)ncc2c(n1)COC2 N1(C(C2CCS(=O)(=O)N2)=O)CCC2(CCCN2c2cnc(F)cn2)CC1 c1(C(N(C2CCN(C(c3[nH]c(O)nc3C)=O)C2)CC)=O)cccn2ncnc12 CC1(C)CC2(CCN(C3CCC4CC3CN4C(c3cnoc3)=O)C2)CO1 N1(C(COC2(C#C)COC2)=O)CCNC(=O)CC1C.C1C(O)CC(=O)N1 CCCCCCC(=O)N(CC)CC1CCCN(C(c2ccnn2CCOC)=O)C1 Cn1cnn(CCNC(=O)C(CC2CC2)NC(c2cc(C(N)=O)[nH]n2)=O)c1=O C(C)(C)(CC(=O)N(CCNC(C1CC(=O)C1(C)C)=O)CCOC)SC c1(C(N2CCC3CN(C(=O)CC4CCCCCC4)C3C2)=O)cnc2n1CCOC2 c1(C(c2nnnn2C2CC2)NC(c2ncc(C)s2)CC)ccc2c(c1)OC(F)(F)O2 N1(C(c2n[nH]c(C)c2Br)=O)CCN(C(c2cn(C3CC3)cn2)=O)C2CCC12 c1(C(C)C)nc(C(=O)OC(C)(C)C)c(NC(=O)OCC2C3CCCCC23)s1 CC1CCCN(C(=O)C(F)=CC2CC2)C1CCNC(=O)CNC(C1CCC1)=O C(CCCCC(=O)N1CCCC1CCCNC(=O)C(O)CSC)OC c1(C(N2CCC(NC(C3C(F)(C(=O)OCC)C3)=O)CC2)=O)cnc(OC)c(Cl)c1 N1(C(CCCSC)=O)CCCC(C)(C)C1C(=O)NCc1ccnc(C#N)c1 N1(C(C(C)CC2CCCCC2)=O)CCC(C(C)NC(c2cnns2)=O)CC1 c1(C(N(CCCNC(c2nncc(OC)c2)=O)C(C)C)=O)ccn2cncc2c1 N1(C(=O)OC(C)(C)C)CCOCC1(C)c1cn(C2C=CCCC2)nn1.C1(=O)CO1 C(CC(C)C(=O)NCC(CCCC)NC(=O)C(C)=CC1CC1)=CC C1(CCC#C)(CC(=O)N(CCC)CCNC(=O)CC2OCCC2C)OCCO1 C1(NC(C(C2C(C)(C)C2(C)C)=O)=O)CCCC(NC(c2ccc(CO)o2)=O)CC1 N1(C(c2c(CC)oc(C)c2)=O)CC2CC(C)N(C(=O)Cc3cnsc3)C2C1 CC(C)(F)CC(=O)NCC12CC1CN(C(=O)C1CC1)C2 c1(CNC(=O)Cc2ccnn2C2CNC2)ccccc1I c1(C(=O)NCCC(=C)CNC(=O)C(N2CCOCC2)C)c(C)nsc1Cl C12(C(=O)NCCOCCOCCOC)CCC1C2.C1C(=O)N1.C1(S)CC1C C1(C2(C)N=N2)CCN(C(=O)CC2CCC(C#N)C2)CC1 Cc1cc(Cl)c(C(=O)NCC(C)(C)NC(=O)C2=CCCS2)cc1Br N1(C(C2C(C(=C)C)OCC2)=O)CC(NC(=O)C2=CCC2)CC(F)(F)C1 C1(C2CC2)(NC(CN(C)CC)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)C1 C1(NC(C2CC(C)OC2)=O)(CNC(C2CCN(C(C)C)CC2)=O)CCOCC1 N1(C(C(C)NC(C)=O)=O)CC2CN(C(c3cc(F)ccc3Cl)=O)CCC12 c1(C(N2CCCC(c3ccnn3C)C2)C(=O)NCCOC)c(Cl)c(C)nn1C C(=O)(C(C)S(=O)(=O)C(C)C)NCc1cccc(CNC(CSCC#C)=O)c1 CC(CCC(F)(F)F)NC(C1(NC(=O)C=CC2CCCCC2)CSC1)=O c1(C(=O)NC2CCC(CN(C(C(C(C)C)F)=O)C)CC2)cnc2ncnn2c1O N1(C(c2c(CC)ocn2)=O)CCC(c2cn(C3CCCN(C)C3)nn2)CC1 S(=O)(=O)(c1cc(C2(C)OCCO2)ccc1F)NCc1cnn(C)c1C(F)F C1CCN=C2C=C(N=CN2)O1.CCC1C(=O)N1.c1(NC(=O)OC)ccccc1 c1(C(N2CCOCC(C(C)C)C2)C(=O)NC(C)(C)C)ccc2nonc2c1 C1(C(N2CCOC(CC3CC3)C2)=O)CCOCCN1C(c1n[nH]c2c1COC2)=O Cc1noc(C)c1C=CC(=O)NCCC1CSCCN1C(c1sccc1C#N)=O C1(CCC)CN(C(c2cnccc2Br)=O)CCN1C(c1cccs1)=O c1(OC(COC)C(=O)Nc2ccn(CC)n2)ccc(Cl)cc1C.C12CC1C(=O)N2 C1(NC(C(C(C)C)n2cc(C)nc2)=O)CCCN(C(c2ccco2)=O)CC1 CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CCOCC1CNC(=O)C=Cc1ncco1 CCC(C)(C)C(O)C(=O)NCC1(OC)CCN(C(c2c(Cl)nn(C)c2Cl)=O)C1 N1(C(CN(C)C)=O)CCC=C(C(=O)N(CC(N)=O)C)C1 Cc1oc(C)c(C(N2CCOC(C(=O)NCC(C)C(C)O)C2)=O)c1C N1(C(COc2ccc(C(=O)OC)cc2)=O)CC(NC(C2CCCO2)=O)CCC1C C1(OC)CN(C(c2cncnc2)=O)CC1C(=O)N(CC(C)C(C)C)C c1(C(C(=O)NC2C(C)N(C(C3CCC3)=O)CC2)O)ccc(Cl)c(F)c1 c1(C(=O)NC2CC(CC(=O)NC3CC(=C)C3)C2)cnn(C)c1C N1(CC2(NC(c3cscc3Cl)=O)CC2)CCN(C(C2CC(F)(F)C2)=O)CC1 CON=Cc1ccc(C(=O)NC2CC3CC2N(C(C2C(C)C2C)=O)C3)cc1 N1(C(CC(OCC)OC)=O)CC(NC(c2cccn2CC)=O)CC(F)C1 Cc1ccccc1-n1nc(C(C)O)nc1CN1CCC(C)C1 c1(C2N(C(=O)NC3C(c4ccc(=N)[nH]c4)CCC3)CCC2)cc2ccccc2o1 CCC(C)C(C(=O)NC1CC(C(=O)N(C2CCCC(C)C2)C)C1)OC c1(OC)c(C(N2CC(C3(NC(=O)C(C)c4cc[nH]n4)CC3)C2)=O)ccnc1Cl C1(CCC(=O)N(CCC#C)C)CCCN(C(c2ccccc2C2CC2)=O)C1 N1(C(C2C(CCOC)C2)=O)CCCC12CCCN(C(=O)NC1CCC(C)(C)C1)C2 C12(NC(C(C)=CC3CC3)=O)CCC(CN(C(=O)Cc3ccccc3)C1)C2 C=C(C)CCCC(=O)NC(C(=O)NCc1ccc(C)cn1)c1cccs1 c1(OC)cc(C)c(C(=O)NCC2(NC(=O)CC(C)(C)C#N)CC2)c(C)c1 CC(CC(=O)N1CCC(n2cc(CNC(=O)C(C)N(C)C)nn2)CC1)C(C)(C)C C1(C(N2CC(C)C(NC(C34CC3COC4(C)C)=O)C2)=O)CC2CC(O)CC(C1)C2 CCCCCC(F)C(=O)NC(CCC)C(=O)NC1CCOC1C c1(C(=O)NC(c2ccccc2)C)ccc(Cn2cccn2)o1 N1(C(C2(N(C)C)CC2)=O)CCCC(O)(CCNC(=O)COCCCN=[N+]=[N-])C1 C1(CCCc2ccccc2)C(=O)N1.c1(C(C)CC2(CC)COC2)cccc(F)c1 C(C1CCCN1C(C1CCCN1C)=O)=CC(=O)NCC(C)NC(=O)OC O=C(C1=CC2CCC(C1)C2)NC1CC(NC(C2Cc3ccccc3N2)=O)C(O)C1 c1(CN2CC(NC(C(CC)c3ccccc3)=O)C2)ccccc1Br c1(N2C3CC(CNC)CC2CCC3)nc2c(c(=NC(C)CNC(C)=O)[nH]1)SCC2 Cc1occ(C(F)(F)F)c1C(N1CC(NC(=O)Cc2cccc(O)c2)C(O)C1)=O N1(C(C=CCN(C)CC)=O)CCN(C(=O)C=CC2CCCCCC2)CC(O)C1 C12(NC(C3CC(F)(F)C3)=O)CCCC1N(C(=O)COCCOC1CCCC1)CC2 CN1CCCC(CC(=O)NC2COCC2CNC(=O)C=C(Cl)Cl)C1 C(C)(C)(CC(=O)NCCn1ccnc1)N(C(C1C(C(C)C)OCC1)=O)C N1(C(c2cc(C)ncc2C)=O)CCN(C(c2ccnc(Cl)c2N)=O)CC(O)C1 C(CC1CCC1)CN=c1[nH]c(N2CCC3C(C2)C3(F)F)nc2c1CCC2 C(CC(C)CO)NC(C(C1(O)CCC1)NC(C(C)OCOC)=O)=O N1(C(C2C(=O)NCCCC2)=O)CC2CC1CN(C(C1CC3CCC(C1)C3)=O)C2 c1(OCC)ccc(CC(C)C(=O)N2CC(c3ncc(Cl)s3)C2)cc1 C1(CC)CN(C(C2CCCCS2)=O)CCN1C(=O)CC1CC=CCC1 C1(C)(NC(c2ccc(C)n2C)=O)CCCN(C(C2(C#N)CCCO2)=O)C1 C1(C(N(C2CCCN(C(C3C(C)CC3)=O)C2)CC2CC2)=O)CC12CCCCC2 c1(C(N2CCC(C3CC3)(NC(CSC)=O)C2)=O)cncc2cccnc12 C(CCC(=O)N1CC(C(N)=O)(OCC)C1)OCC(=C)C C1(NC(c2ccc(C)nc2C)=O)CC2CCC1CN2C(c1cc(N)nc(Cl)c1)=O c1(NC(CC2N(S(C)(=O)=O)CCC2)=O)nc[nH]c2ncc(Br)c1-2 N1(C(COCC(=O)OC)=O)CCC2(CCOCC2)C(CNC(=O)C(F)OC)C1 c1(C(CO)NC(C2(CC=C)CCOC2)=O)ccc(Cl)cc1Br C1(C(=O)NCC(CNC(c2cnc(CCC)s2)=O)O)Cc2cccnc2C1 C1(NC(c2c(C)n(CCO)cc2)=O)CN(C(C2(C#N)CC(C)C2)=O)CCC1(C)C C(=O)(C1=NNC(=O)CC1)N1CC(COC)N(C(C2CCOC2=O)=O)CC1 c1(CC(=O)NCCc2csc3ncsc23)cc(F)c(O)cc1F C(=O)(CCCC(=O)N1CCCC(CO)(NC(=O)CCCC2CC2)C1)N(CC)CC C1(CC(N2CC(F)(F)C2)=O)C2CCCC2N1C(=O)C=Cc1cnccn1 C#CCC(C)(C(=O)NCC(F)(F)COC)NC(=O)C#CC1CC1 N1(C(c2c(C)occ2)=O)CCC2CN(C(=O)C=Cc3nnn(C)n3)C2C1 C(=O)(C1=COCCC1)N(C(C(=O)NC(CCCCC)C1CC1)C1CC1)C C(=O)(CC(C)C(C)C(C)C)NC(CC(C)C)CNC(c1c(F)cc(F)cc1F)=O c1(CCC(=O)NC2C(CNC(C(CCCOC)C)=O)C2)ccc2ccccc2c1 C1(CCCCCC2CC2)CCNCC1.[nH]1cc(-c2cnccn2)nn1.O=C1C2CC1C2 C1(C(=O)NC2(CNC(=O)COCC3CCOC3)CCC2)C2CCOCC12 Cc1cc(C(=O)NCCC2CN(C(=O)C(F)(F)C(F)F)CC2C)c(C)cn1 c1(CC)nonc1C(=O)N(C1CCN(C(c2cnn(CC(C)C)c2)=O)C1)CC N1(C(C(CCOC)OC)=O)CCN(C(=O)CCc2ccco2)CC1C1CC1 Cc1c(C(N2CCC(c3cn(CC4CC4)nn3)C23CC3)=O)cccc1Cl c1(C(N2CC3C(NC(CC(C)C4CCCCC4)=O)C3C2)=O)cccc(S(C)=O)c1 c1(CCC(=O)NCC2N(C(C(CC)C)=O)CCC2)cccc(C(=O)OC)c1OC Cc1ccc(C(N2CCCC2C2(NC(C3CCCN(C)C3)=O)CC2)=O)c(Cl)c1 C(CC(=O)NCc1nc(C#N)cs1)(C(C)C)NC(C1ON=C(C)C1)=O c1(-c2ccc(Cl)c(Cl)c2)cc(=NC2CC3CCC(C2)S3)[nH]c2ncccc12 c1(C(C(=O)N(CC(CC)NC(CNC(CC)=O)=O)C)CC)ccc(F)cc1 c1(C(N2C(CC(c3n(C)cnc3)=O)CCC2)=O)ccc(S(N)(=O)=O)cc1 C1(C(N(C(CC(CC)C)C)C)=O)C2CCC(C2)C1NC(C1(COC)COC1)=O c1(C(NOCC(=O)N(C)CCNC(C2OCCC2C(F)(F)F)=O)=O)cn(C)cn1 Cc1ccc(C(C)(C)CC(=O)N2CC(N(C)C(c3cccnc3CO)=O)C2)cc1 S(=O)(=O)(c1ccc(Cl)s1)N1CCN(S(CCOCC)(=O)=O)C2C1C2 C1N=C2NC(=NCC(CCSC)C=CC3=C(N=C1)CCC3)NC1=C2CSC1 c1(C(N2CCCC(CCNC(C3C(C)CCC3)=O)C2)=O)cc(Cl)ccc1Cl CC1CN(C(c2cccnc2S)=O)CCN1C(c1cc(Cl)c(Br)cn1)=O c1(N2CCC(NC(c3c(C)oc(Cl)n3)=O)C(C)(C)C2)nc2cc(Br)cnc2s1 N1(C(C2CN(CCC)C(=O)C2)=O)CCCN(C(=O)CNS(=O)(=O)CC)CC1C N1(C(CC2C(C)CCC2)=O)CCCN(C(c2ncsc2C2CC2)=O)CC1 C(=O)(C1=NOCC1)NC(CN(C(c1cccc(C2CC(F)(F)C2)c1)=O)CC)C c1(C(=O)NC2CCN(C(c3n[nH]c(C)c3F)=O)C2)nsc2ccccc12 c1(OCC)ccc(C(=O)N(CCNC(C2CC2(Cl)Cl)=O)C2CC2)cc1OC.OC C1(C(=O)NC2COC2)CCn2ccnc2C1.C1(=O)C(C)N1CCCSC C1(CNC(Cn2cc(CNC(CC3(OC)CCC3)=O)nn2)=O)CCN(C)CC1 N1(C(c2ccc(CNC(c3c(C)ncs3)=O)cn2)=O)CC(C)OC2(CCC2)C1 C1(C(N(CCCC)CCOC)=O)CC12CC(NC(C1CCC(=O)O1)=O)C2 N1(C(C(COCC)C)=O)C2CCC(C(=O)NCc3ccc(F)c(F)c3)C1CC2 O=C(C1CCCc2nncn21)NC12CCCCC1CN(C(C1CC=CC1)=O)C2 c1(C(N(C2(CC(=O)NC3CC(=O)C3)CC2)C)=O)ccc(O)c(Br)c1 C1(NC(CCCc2scc(C)n2)=O)CCN(C(=O)C(=O)NCC2CC2)CC1O CCCCC(CCC)NC(c1conc1C(C)NC(=O)Cc1ccsc1C)=O C1(C(=O)NCCN(C(=O)CCS(C)(=O)=O)CCOC)CCC2(CCOCC2)C1 N1(C(c2ncc(C)c(C)c2)=O)CC(C)(C)OC2(C1)CN(C(=O)Cn1nccn1)C2 c1(SC)ccccc1CC(N1CC=CC1NC(=O)CC1CCOC1(C)C)=O C(CC(O)CC(=O)N1CCC(CN(C(=O)CNC(=O)C2CC2)C)C1)SC C1(CCNC(=O)CC2(CNC(c3cccc(=O)o3)=O)CC2)CCCNC1=O Cc1ccc(C(N2CCC(O)(CNC(c3scnc3C(C)(C)C)=O)C2)=O)nc1C c1(C(=O)NCC(=C)CCNC(C2CC2[N+](=O)[O-])=O)noc2c1CC(F)(F)CC2 C1(NC(c2nc(C(C)NC(=O)CN3CC(C)(C)C3)oc2)=O)CCCC1(C)O C1(CC)(NC(=O)C=Cc2cccc(CO)c2)CCN(C(=O)CCN(C)CC)CC1 C(CCN=C(NC(C)COC(C)OC)N1CCC(F)(F)C2(CC2)C1)OC C1(NC(c2cc(C)ns2)=O)CN(C(c2cncnc2C(C)C)=O)CCC1C c1(C(=O)NCC(CC)(C)NC(C2CC(F)C(=O)N2)=O)oc(C(C)C)nc1C Cc1ccc(O)c(C(=O)NCC2CC(C(F)(F)F)CN2C(=O)CCC2CC2)c1 C1(NC(C(CC)CC)=O)COCCN(Cc2ccccc2F)C1 C1(NC(=O)CC2CCOCC2)CC2CCC(C1)N2Cc1ccccc1Br c1(N(C(C)C2CC2)C(=O)NC(C)CO)cccc(C#N)c1 C(CCC(C)NC(C1(SC)CN(C(c2coc(OC(C)C)n2)=O)C1)=O)=C(C)C c1(NCCN(C2CC2)CC)ncccc1S(=O)(=O)N1CCOC(C#N)C1 C1(C(=O)NCC2CC(NC(c3scc(C)c3)=O)C(O)C2)CCCC(F)(F)C1 C(C)(CN=c1ccc(Cl)c(C)[nH]1)OC(CC)(C)C N1(C(c2c(CC)c(OC)ccc2)=O)CCC2(C1)CN(C(=O)CC(C)C)C2 CC1COc2c(C(=O)NC(C)(C)CNC(C34CC(C)C3C4)=O)cnn2C1 C1(NC(C(C)OCOC)=O)CC(F)CN(C(C2CC3CC3C2)=O)C1 N1(c2c3ccc(C#N)cc3ncc2)CCC2(CC1)OC(=O)Nc1ccc(F)cc12 C=CCC(C)(CC)C(=O)NC1CC2CC1N(C(c1cncc([N+](=O)[O-])c1)=O)C2 Cc1ccc(C(N2CC(C(F)(F)F)CC2CNC(=O)CC(C)F)=O)c(F)c1F C(=O)(C1CC=Cc2ccccc21)NCC#CCNC(c1cnc2scc(C)n21)=O CC1C(=O)N(CC(N2CC(CNC(C3CC(O)C3)=O)CCC2C)=O)C(=O)C1C c1(OC)nccc(C(=O)NCC2CC2CNC(c2cccc[n+]2[O-])=O)n1 N1(C(C2C(=C)C2)=O)CCCCC1CNC(=O)Cc1cncc(C)c1 CCC(CNC(=O)COc1cc(C)on1)N=c1nc2[nH][nH]cc-2c(O)n1 C(C(O)CC(=O)NCCc1ccccc1O)NC(C1(C)CSC1)=O c1(C(CO)NC(c2cc(-c3csc(CO)n3)c[nH]2)=O)cccc(Cl)c1 C=CCC(C(=O)N1CC(NC(c2cnc(C(C)(C)C)o2)=O)C(C)C1)C(C)C CCCC(C(O)C(=O)N1CCCC(O)C1C)NC(=O)C=Cc1cccnc1 C1(NC(c2c(C)oc(Cl)n2)=O)CN(C(c2nn(C)nc2C(F)(F)F)=O)CC1(C)C C1(C(=O)NC2(COCC)CC2)CCCCCN1C(=O)CNc1ccccc1 N1(C(C23CC(C)(C2)C3)=O)CC2=C(C1)CN(C(c1ncccc1F)=O)C2 N1(C(C(C)(C)CF)=O)CCC(NC(c2cc(C3CC3)ccc2F)=O)C(CO)C1 c1(CC(=O)NC2CCOCC2NC(C2CCCC23CC3)=O)ccncc1Cl c1(OCC(=O)NC(C2C(C(=O)NCCC(C)(C)OC)C2)C)ccc(Cl)cc1 C(N=c1[nH]c(=NCC2COC(=O)O2)c2ncccc2[nH]1)c1ccc(C(C)(C)C)cn1 Cc1cc2nc(C(=O)NC3CCN(C(=O)C4=CCCOCC4)C3)cn2cc1C C1(NC(c2ccc(OC)s2)=O)CN(C(=O)COc2cccc(F)n2)CC2CC12 N1(C(c2c(C)nsc2)=O)CCCN(C(c2csc3ccccc23)=O)CC1C(C)C N#Cc1cccc2c1CCN(Cc1cccc3c1OC(F)(F)O3)C2 c1(C(=O)NCC(CNC(C2C(CCC)C2)=O)F)sc(=N)[nH]c1-c1ccccc1 Cc1ccc(O)nc1NCc1ncc(-c2ccc(Cl)cc2)o1 C(C)(CCN=c1nc2sccc2c(NC2C=CC=CC=C2)[nH]1)OC C1(NC(c2nn(CC)c(C3CC3)c2)=O)C2CC1N(C(=O)CCC(C)C)C2C Cc1cc2sc(C(=O)NCCC3(O)CN(C(=O)CCCC4CCC4)C3)cc2s1 CCC(CCC(C)C)(c1nnnn1C1CCC1)NCc1ccccc1OC c1(OC)c(C)cc(C(N2CC3(CNC(C4SCCS4)=O)CCC2CC3)=O)cc1C N#Cc1c(F)cccc1S(=O)(=O)NC(=O)CCOCC1CCC1 c1(C(N(C)CC2CCN(C(CCCOC)=O)C2)=O)ncccc1Br c1(C(N2CCCC2CS(N)(=O)=O)=O)sccc1C=O.N1CCCC1 CC(C)(F)C(C)(F)C(=O)N1CC2CCC1CC2NC(=O)CC1CNC(=O)O1 N1(Cc2ncc(CC)o2)CC(c2ccccc2)C(F)(F)C1.C1CNC(=O)N1 C1(NC(CN(C2CCSC2)C)=O)CCCCC1CNC(=O)CC1(O)CCOC1 N1(C(c2ccc(C3CC3)cc2F)=O)CCN(C(C2(O)CCSCC2)=O)CC1CO N1(C(c2c(C)ocn2)=O)CCC(CNC(c2c(F)cccc2Br)=O)C(O)C1 C1(NC(CCCC(=O)OC)=O)C2CCCN(C(c3[nH]ccc3C)=O)C2C1(C)C c1(CC)c(C(=O)NCC(C2CCCC2)NC(=O)C(C(C)C)C2CC2)nnn1CC c1(COCC)cccc(C(N2CCC(CN(C(=O)Cc3csnc3C)C)C2)=O)c1 N1(C(C(COC)(C)O)=O)C2CCC(C2)C1C(=O)NC1CCCC1C#N N#Cc1cc(N2CCOC(c3cccs3)C2)c2ccccc2n1 c1(OC)c(NC(=O)CN(C(=O)CNC(C2CC2C)=O)CC2CC2)cccc1C CC(C)C(C(=O)N1CCCN(C)CC1)C(C)NCC(=O)Nc1cccnc1 C(=O)(CS(=O)(=O)C1CC1)N1CC(NC(c2c(C)nn(CCC)c2C)=O)C(C)CC1 CC1(C(=O)NCC2CN(C(=O)Cc3nc4ncccn4n3)C2)CCCNS1(=O)=O c1(OC)cc(F)c(C(N2CCN(C(=O)CC3CC=CCN3C)CC2)=O)c(F)c1 CS(=O)c1ccc(C(N2CCOCC(CNC(c3cc(F)c[nH]3)=O)C2)=O)cc1 c1(C(N(C2CCN(C(=O)C=CSC)CC2)CC)=O)ccnc2c1nnn2C N1(C(C2CN(CC(C)C)C(=O)C2)=O)CC2CC1CN2C(c1ccccc1N(C)C)=O N1(C(C2C(C)CCN2C(=O)Cc2cn(C)cn2)=O)CC2CCC(O)C(O)C12 CC(C)C(C(C)NC(c1cc(Cl)sc1Cl)=O)NC(=O)C=CC1CCCC1 C#Cc1ccc(CC(=O)NCCC(=O)NC(C2CN(C)CCO2)C)cc1 C1(NC(C(C)OCCCC)=O)CCCCC1NC(=O)C(C1CC1)SC c1(C(=O)NC(C2CN(C(=O)Cc3cnsc3)CCO2)C)cccc(C2CC2)c1Cl Cc1ncnc(C)c1CC(=O)NCCCC(C)(C)NC(C1CC2(CCC2O)C1)=O N1(C(c2ncc(Cl)cc2F)C(=O)NC2(C(=O)OC)CCCC2)CC(F)(F)CCC1C C(=O)(CC(C)(O)C(F)(F)F)NC1C(CNC(c2cc(OC)c(C)cc2)=O)C1 CN(C)NC(=O)CCC(=O)N1CCC(CCNC(=O)COCc2ccccn2)C1 C1(C)(CC)CC(C(=O)NC2CC(NC(=O)Cc3ccn(C)n3)C23CCC3)CCO1 Cc1ccn(CCC(N2CCC(CNC(=O)CC3CCC(=O)N3)C2)=O)n1 Cc1cc(C(=O)NCC2(C(=O)NOC3CCCC3)CC(F)(F)C2)cnn1 CCC(CC(=O)NCC12CCC(CN(C(c3nscc3C)=O)C1)C2)C(C)(C)C S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)NC1C(C(=O)NCc2cccc(Br)c2)C1 C(C(=O)N1CCC(C(N2CCOC(CCN(C)C)C2)=O)O1)N(C)C C(=O)(CC(F)(F)Br)NCC1(O)CC(NC(c2[nH]cc(CC)c2)=O)C1 N1(C(C(CC)OCC)=O)CC(NC(C2SCC=C2C)=O)CC12CCCCCC2 C(c1cnn(C)c1)=CC(=O)NC(C1CCN(C(C2CCCC(CF)C2)=O)CC1)C CC1CN(C(C2CC3(CCC3)C2)=O)CC(C(N2CC3CCC3C2)=O)O1 c1(NC2CCN(Cc3scc(C(=O)OCC)c3)CC2)cc(O)ccc1COC C1(C(N2CCC(CCCCCNC(C3C(C)C3)=O)CC2)=O)CC1C1CCOCC1 c1(OC)ccccc1C(O)C(N1CCC(CCNC(=O)CSC)C1)=O C1(C(=O)NC(COC)C2CC2)OCCC1CNC(=O)C(N1CCCCC1)C C1(n2c(C3CC3(C)C)nc(-c3ccc(C)o3)n2)CC(C)OC(C)C1 N1(C(C(=O)NCCSC)c2cnsc2)CCC(CCCN2CCCCC2)CC1 C1(CCC(=O)N(CCCNC(C2(C(F)F)CC2)=O)C(C)C)CCC(O)CC1 C(=O)(C(F)C(C)(C)O)N1CC(NC(CC(C=C)C)=O)C(c2ccc(OC)cc2)C1 C(=O)(C1=C(Cl)CC1)N(C(CNC(=O)CO)C(N1CCN(C(C)=O)CC1)=O)C C1(SCC)CN(C(c2cnn(C)c2CC)=O)CC1C(=O)N(C(C)C(C)C)CC c1(C(=O)NC2C(OC)CN(C(c3cnnn3C)=O)CC2)c[nH]c2ncc(F)cc12 C1(C(=O)NC2CCCC2C(=O)NC(CC2CCC2)CO)CCC(F)(F)C1 N1(C(CSCC#C)=O)CCC(CO)(CNC(C2CC2C(C)(F)F)=O)CC1 C(CCCCC(=O)NCC(C)CC(=O)N1CCC1C(C)O)=CC CCCCCCCC(C)Cc1nc(CC2CCCC2)nn1-c1cccnc1C C1(C(N2CC(NC(c3cc(C)oc3)=O)(CO)C2)=O)CC(O)CN1C CCC(C)(COC)C(=O)NC1CCCC1NC(=O)C1=CCCC1C c1(C(C)C(=O)NC(C(=O)NCC(n2ccnn2)C)C2CCOC2)ccnn1C c1(C(=O)NCC2CC(N)C(O)C2)cc(OC)cc(Cl)c1.C1(CC(=O)C2CC2)(OC)CC1 c1(N(CC=C)C)nccc(=NCC2CCn3ccnc3C2)[nH]1 c1(OC)cc(C(=O)N(CCCNC(C2CN(C)C2)=O)C)cc(Br)c1OC CC1CCN(CC(=O)N(C(=O)C(O)CC2CC2)Cc2ccccc2)CC1 C1(CC(=O)NCCN(C(=O)CCCc2cccs2)CCC)COCC(C)O1 C(CCCCC(=O)NC1CCOC(C(C)C)C1)NC(c1nc(CCC)oc1)=O Cc1cc(C(N2CC(NC(=O)Cn3ccc([N+](=O)[O-])n3)C3CC23)=O)nnc1O CCC(CN(C)C)C(=O)NC(C)CNC(=O)CCc1cccc(Br)c1 N1(CC=C)CC2CCC(NC(c3nccc(C(C)(C)C)n3)=O)CC2C1 CCCC(CC1CCCC1)C(=O)NCc1cccc(-n2cc(CCO)nn2)c1 N1(c2ccnc(SC)n2)CCC2(CCN(Cc3cccc(Cl)c3O)CC2)CC1 c1(C(N2C(CNC(C3(C#C)CCCC3)=O)CCC2)=O)nc(C)c(C)cc1Br C1(C#N)(C(=O)NCC2CC(NC(C=Cc3cncc(C)c3)=O)C2)CC12CCCC2 CN1CC(F)(CNC(C2CC(C)(NC(=O)COC3CC=CC3)C2)=O)C1 c1(CCC)sc(C(=O)NC2(CNC(C3(CF)CC(=O)C3)=O)CCOC2)cc1CC C(N=c1[nH]c(N2CCC3CC3C2)nc2c1CSC2)C1(OC)CC1 C1(C(N2CC(OC)(CNC(=O)CCc3ccccc3)C2)=O)CCCC(O)C1 CCC(C)CCC(O)CC(=O)NCC(C(C)C)NC(=O)CN1CCC(CO)CC1 C1(NC(=O)Cn2cccn2)CC2(CCN(C(C3CC4(C3)CC4(F)F)=O)CC2)C1 c1(NC(C)CCNC(C2(c3cc[nH]n3)CC2)=O)c(C#N)cccc1[N+](=O)[O-] C1(CNC(C(=O)NCC2CCCC(F)(F)C2)=O)CCCCC12OCCO2 Cc1ccc(C(N2CCCC2(C)CCC(=O)N2CC(N3CCC3)C2)=O)c(O)c1 n1(CCNC(C2C(C)CC2)=O)cnc(C(=O)NCCCCF)c1 c1(COC)ccnc(C(=O)NCCCC(C)NC(=O)Cc2cc(C)on2)c1 C1(CNC(CCC=C(C)C)=O)CCN(C(=O)CS(=O)(=O)NCC2CC2)C1(C)C C#CC1CN(C(=O)C(C2CCOCC2)C)CCN1C(c1cncc(C)c1)=O C1(n2cc(C(C)O)nn2)CCN(C2CCN(C(C3OCC3(C)C)=O)C2=O)CC1 C1(CNC(c2c(C)nn(CCO)c2)=O)CCN(C(=O)Cc2csc(S)n2)CC1C N1(C(C(C)OCCC(C)C)=O)CCOCC1CCNC(C12CC(CO1)C2)=O C1(CNC(COC2CN(C(C(CC)(C)N(C)C)=O)C2)=O)CC(C)(C)CCO1 c1(C(C)=O)cccc(C(=O)NCCC(C)(C)NC(c2cc(C(N)=O)[nH]n2)=O)c1 C(C(=O)NCc1cn(CC(=O)NC(C)C(OC)OC)nn1)(C(C)(C)C)NC c1(C(c2n(CC)nnn2)NC2CC(Cc3ccco3)C2)cc(C(N)=O)ccc1F C(C(=O)NOC1CC1)(C1(C)CC1)NC(CC1CC(=C)C1)=O C1(NC(CC2ON=C(C)C2)=O)(CNC(=O)C(n2ccc(C)n2)C)CC(F)(F)C1 N1(c2sc3ccn(C)c3c2)CC2CCC(C1)N2Sc1[nH]cc2c1CCS2(=O)=O Cc1cc2sc(C(=O)NC(C)CCCNC(c3cccc(Cl)c3F)=O)cc2s1 C1(C(N2C(C3CCN(C(c4n(CC)cnn4)=O)C3)CCC2)=O)C2CC3C(C2)C13 n1(C(C)(C)C)ncc(C(=O)NC2(C)CC(NC(C3CC4CCC34)=O)C2)c1Cl Cc1occ(C(F)(F)F)c1C(=O)NCCC(O)CNC(=O)CCCNC(N)=O C(C)(C)(C(C(=O)OC)NC(c1nc(-c2ccc(Cl)c(F)c2)cs1)=O)OC C(=O)(C1CCS(=O)(=O)c2ccccc21)NCCN(C(=O)COC(F)F)C C1(C(N2CC(C)(O)C2)=O)(N(C(=O)CC2CCCC23CC3)C2CC2)CCC(C)(C)C1 C=C1CC2(C1)CC(C(=O)NCC1(C)CCN(C(C3CC(S(C)(=O)=O)C3)=O)C1)C2 c12cccc(c1O)C(=O)N2.C12(C(N(CC(C)N3CCC3)CC)=O)CCCC1C2(F)F C1(O)(CNC(C2(C)C=CCC2)=O)CCCN(C(c2cn(CC(N)=O)nn2)=O)C1 C1(C(C)(F)F)CCCN(C(=O)C=CC(=O)NCc2nnc(Sc3nc[nH]n3)o2)C1 c1(C(=O)NCC(CNC(=O)C(O)CC2CCCCC2)CO)c(F)cc(F)cc1F Cc1cnnc(C)c1C(N1CC=CC(C(N2CCOC(C)(C(C)C)C2)=O)C1)=O CC1CC(=O)NC(C(=O)NC(CNC(=O)C(C)NC(=O)C2CC2)C2CC2)C1 c1(C(=O)NCCN(C(=O)C=Cc2cnccn2)CC)cnc(C(F)F)cc1C c1(C(CC)(C)NC(C2(c3noc(C(F)(F)F)n3)CC2)=O)ccccc1OC(F)F C1(C)(NCC(=O)NC(CCN(C(=O)C(C)(C)C)C)c2cccs2)CCCCC1C c1(CC(=O)NCC2CN(C(C(CC)(C)OC)=O)CC2O)ccc(Cl)c(F)c1 Cc1nc(C(=O)NCC(C)NC(C2CC23CC3)=O)ccc1Br C(=O)(C1=C(Cl)CCOC1)N1C(CN(C(CCCOCC)=O)C)COCC1 c1(C(N2C3CN(C(CC(C)C(F)F)=O)C(C3)C2)=O)ccnc2ccnn12 N1(C(C2(NC(C(C)Cn3cccn3)=O)CCOCC2)=O)CC2CCC2(CO)C1 C#Cc1cc(F)c(C(=O)NC2CCSC23CN(C(=O)CC2CCOC2)C3)cc1F N1(C(C(C)(C)C)=O)CCOC(CNC(C2CCC2(F)F)=O)C1 N1(C(c2cnc(C3(CC)CC3)o2)=O)CCC(n2cc(C(=O)O)cn2)CC1 c1(CCC(=O)NC(CNC(C2(CCOC)CC2)=O)C)nnc(C)n1C CCC(C)(C)CCCC(=O)NCC1CC(NC(c2ccc3cc[nH]c3c2)=O)C1 C(CC1CCOCC1)(C(=O)NOCC(F)(F)F)NC(c1ccc(C)nc1)=O C1(CN=C(NC(C)CF)NCC2(CC#N)CC2)CC(C)(C)CC(C)(C)C1 C(=O)(C(=O)C(C)N1CC(CC(F)(F)F)C(OC)C1)OC c1(CC2(F)CC(CNC(=O)NC(c3ccsc3)CC)C2)cc(O)ccc1C N1(C(C)C(=O)NC(Cc2ccc(F)cc2)CO)CCOCC(NC(C2CC2)=O)C1 Cc1cccc2oc(C(=O)NCC3(F)CC(NC(c4ccncc4)=O)C3)cc12 N1(C(C2C(CC(C)(C)C)C2)=O)CCN(C(=O)C2=CCOC2)C(COC)C1 c1(C(=O)NC2C(NC(c3nn(C)c(C(F)F)c3)=O)COC2)cnc2cccnn12 C(C(CNC(=O)C(F)C1CCC1)S(C)(=O)=O)NC(c1[nH]cc(C)c1)=O c1(C(N2CCN(C3CN(C(C4(C)C=CCC4)=O)C3)CC2)=O)nc2ncccn2n1 N1(C(c2c(C)nc(O)s2)=O)C(C(=O)NC(c2n[nH]c(CO)n2)C)CC2CCCC12 C(=O)(C1(C)CCCc2ccccc21)NCC1C(NC(C2(C(C)C)CC2)=O)C1 N1(C(CC2N(C(C)C)CCC2)=O)CC2CC(C(N3CCC(O)(CO)C3)=O)(C2)C1 C1(C)(CNC(CSCC#C)=O)CC(F)(F)CN1C(c1cn(C)ccc1=O)=O Cc1ncc(N)cc1C(=O)NC1(CNC(=O)CCNC(=O)CO)CCOC1 c1(CC(=O)NCC2N(C(CC=C)=O)CCC2C)csc2sc(CC)cc12 CC(C)CC(C)CC(=O)NCC(CC(C)C)NC(=O)CCC1CC1(C)C CC(CCCCNC(C1CC(C#N)C1)=O)NC(c1nnn(C)c1C(F)F)=O C1(C(=O)NC2CCC(NC(CCc3n(C)ccn3)=O)CC2)CCC2C(C1)C2(F)F CCCC(C(=O)OC)C(=O)N1CC2CC(NC(=O)CCC(C)C)C2C1 Cc1cncc(C)c1C(=O)N(C(C1CCCN1N1C(C)(CC=O)CC1)C)C C12(C(N3CC(OC)(CNC(C4COC(=O)N4)=O)C3)=O)CCCC(=O)N1CCC2 Cc1ccn(CCC(=O)NCCCN(CCCCNC(C2CC2(C)CF)=O)C)n1 N1(C(CCCSC)=O)CC(C(=O)NCCCC2CC2)C2(CCC2)C1 CN(C1CN(C(C2CCCCC2)=O)CCc2ccccc21)C(C1CNC(=O)C1)=O CCC(CC)(CC)C(=O)NC(CNC(=O)Cc1ccc(O)c(C)c1)CO Cc1cc(C(=O)NC2CCC(NS(=O)(=O)C(F)(F)F)C2)cc2c[nH]nc12 N1(C(C(N2CCOCC2=O)C)=O)CCC(CNC(C2CCC2C)=O)C12CC2 CC1(C)CC(NC(=O)COC2COC2)CN(C(c2cc(Br)n[nH]2)=O)C1 Cc1c(Cl)sc(Cl)c1C(=O)NC(C)CCN(C)C(c1cnn(C(C)C)c1N)=O C1(F)(CNC(=O)C=CCCc2ccccc2)CCN(C(C2(CCF)CC2)=O)CC1 CCC(C)C(O)C(C)C(=O)N1CC(C)(C)CCC1CNC(=O)C(F)C(C)(C)O n1(CC)nc(-c2ccccc2)nc1-c1ccc(CC(F)(F)F)cc1 n1(CC(=O)NCCN(CC(C)O)C(=O)Cc2cc[nH]n2)cnc(C#N)n1 c1(C(=O)NC2CCCN(C(CSc3n[nH]c(=N)s3)=O)C2)cccc2nncn12 C(C(F)(F)C(=O)NC1C2CC1N(C(C1CCCOC1C)=O)C2)OC N1(C(c2cn[nH]c2)=O)CC2C(C(F)(F)F)C2C1.C1(N)COC1 C1(NC(CCc2onc(CC)n2)=O)COCCC1NC(c1ccn(CC)c1C)=O c1(C(=O)OCC)ccc(N2CCN(C)CC2CNC(c2cocc2C)=O)nc1C N1(C(c2ccc(C)n2C)=O)CCCC2CCN(C(=O)CC34COCC(C3)C4)CC12 N1(CC(CC)OC)CC2(CN(C(=O)C(CC)c3ccccc3)CCO2)C1 O=C1NCCOC2=C1C1=CC=CC(=C2O)N(CC(O)C(O)CO)C1=O c1(C(=O)NCC2CCCN(C(CCC#CC)=O)C2)c[nH]nc1[N+](=O)[O-] C=CCC(C)(CC)C(=O)N1CC2CCC(NC(=O)C(C)(C(C)C)NC(C)=O)C2C1 C(=O)(CC(C)CC(C)C)N1C(CNC(CC(CC)SC)=O)CC(C)(C)C1 c1(C(N2C(C)C(NC(C3CCCCN3N=O)=O)CCC2)=O)cc2ccccn2n1 c1(OCC)ccc(C(=O)NCCC2CCN(C(=O)C(C)C)CC2)cc1[N+](=O)[O-] N1(C(CC2(C)CCOCC2)=O)CCC(NC(=O)C=Cc2ncco2)C(F)C1 N1(C(c2c(C)c(O)ccc2)=O)CCC2(CC1)CC(N1CC3CC1CC3(F)F)CO2 Cc1ccc2cc(C(=O)NCCN(C(=O)C(c3cncc(F)c3)C)C)cnc2c1 C1(NC(=O)NCC2(C(F)F)CCC2)(CO)CC2CCC1CC2 CN(Cc1ccc2c(c1)OCCO2)N1CCOCC(CO)C1 CC1(CNC(C2(C)CC2(F)F)=O)CCCN(C(=O)Cc2ccn(C(F)F)n2)C1 N1(C(CCCNC(=O)OCCCC)=O)CC2CC(NCCc3cnco3)CC1C2 c1(C(=O)NCC2(NC(c3nc(C)nn3C)=O)CCC2)ccc2c(c1)C=CCC2 c1(C(=O)NC2(C)CN(C(C3(F)CC=CCC3)=O)C2)cnn2cc(Br)cnc12 CC(C)CC(C)C(=O)N1CCN(C(=O)COCc2nc[nH]n2)C(C2CCC2)C1 C1(CNC(C(C)NC(N)=O)=O)CCN(C(c2cc(Br)co2)=O)CC1 Cn1ccc(C(=O)NCC2CCN(C(=O)CC3CCCC3O)C2(C)C)c(O)c1=O C(=O)(C1=CCC(NC(c2c[n+]([O-])c(C)cn2)=O)C1)N1CC(CC)C(F)C1 c1(CC(=O)NC(c2cn(CC(=O)N(C)C)nn2)CCC)c(C(F)(F)F)coc1C C1(CC)CCN(C(C2CN(C)C2)=O)C(C(=O)NCC2COCC2(C)C)C1 c1(C(=O)NC2C3(CN(C(C(=O)NCC)=O)C3)CCC2)cc(O)c2[nH]c(C)nc2c1 N1(C(CC#N)=O)CC2CC(C1)N(C(c1ccc(F)cc1)=O)C2.c12cccc(c1)O2 N1(C(c2ccccc2F)C(=O)NCCCCCC)CCN(CCN(C)C)CC1C C1(CC(=O)NC(C2CCCN(c3cc(OC)ncn3)C2)C)OCCCC1(C)C C1(C(N2CCC(C(C)(C)O)C2)=O)CCC(NC(=O)CCc2ccc(Cl)s2)CC1 C=C(C)CC(C(=O)N(C)CC1COCCN(C(=O)OC(C)(C)C)C1)N(C)C C=CC1(C(=O)NC(C2CCCN2C(=O)C(C)Cc2ccccc2)C)CCC1 C(=O)(CCC(=O)NCCOCCC(=O)NC(C)Cc1ccncc1)NC C1(CNC(C(=Cc2cccc(Cl)c2)C)=O)CN(C(=O)C(=O)NC2CC2)CCC1C C1(CNC(C2CC2CF)=O)CC12CCN(C(=O)Cn1nc(O)ccc1=O)CC2 N1(C(c2ccc(C(N)=O)[nH]2)=O)CCN(C(C2CCCS2)=O)CC1CO C12(NC(C3C(CC)N(C)CC3)=O)CCC(CC1NC(c1c(C)oc(C)c1C)=O)C2 C1(C)(CC)CC(NC(=O)CCCN(C)CC)CN1C(c1ccc(OC)c(Cl)n1)=O C1(C(=O)NC(c2c(C)n[nH]c2C)C)COCCN(C(C2(C)CC2(C)C)=O)C1 c1(C(N(CC(C)O)CCNC(CCC2N(C)CCC2)=O)=O)cccc(O)n1 CN1CCCCC1C(=O)NCCCCn1cc(C2COC(C)(C)C2)nn1 C1(C(=O)NCCN(C(c2cc(C3CC3)no2)=O)C2CC2)CCC=CCCC1 N1(C(c2ccc(C#C)o2)=O)CCCC12CCCN(C(=O)C(C)CC1CCC1)C2 C(=O)(CCCC(F)(F)F)N(CC(C)(C)CNC(c1cnc(CC(C)(C)C)s1)=O)C Cc1cn2cc(C(N3CCC(O)(CNC(=O)C(F)C(C)C)C3)=O)cc(F)c2n1 c1(OCCN(CC)CC)ccc(NC(C(F)(F)OC)C(=O)OC)cc1OC c12cncc(c1)C(=O)N1C(CCC1)C1(CC1)N(C)C2=O.c1(OCCF)ccn(C)n1 Cc1ccc(C(=O)NCC2CN(C(c3cc(C#N)c[nH]3)=O)CCCO2)c(O)c1C N1(C(CCc2scc(C)n2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)C(C)C1 C(=O)(C1=CC(C)(C)C1)N(C1CCN(CCON)CC1)C(C1CCCCC1)C CN1C(=O)C(=O)N(CC(=O)NCC(C2CC2)NC(C2CCO2)=O)C1=O O=C(NNc1cc(O)nc2ncccc12)NCc1cccc(CO)c1 C1(F)(CNC(C2CCOC2)=O)CCCN(C(C2(C(F)(F)F)CCO2)=O)CC1 c1(CCNC(c2n(CC=C)nnn2)(C2CCCO2)C)ncccc1OC N=c1nc(CC(=O)NCC2(O)CC(C(=O)NCC(O)C(F)F)C2)[nH][nH]1 C#CCCCCCC(=O)N1CCOC(C(=O)NCC2(C)CCCC2)CC1 Cc1c(Cl)c(C(=O)NC(C2CCCN2C(=O)CCC(=O)c2ccc[nH]2)C)nn1C C1(NC(c2nc(C(C)C)oc2)=O)CC2CCC1N2C(c1cnn(C)n1)=O C1(CCNC(C2(CC#C)CCCO2)=O)CN(C(C2CC=CC2)=O)CCO1 C1(NC(c2cncc(SC)c2)=O)CC2(CCN(C(c3n[nH]cc3Cl)=O)C2)C1 C12(C(N(CCC)CCNC(c3cnc(C(F)(F)F)s3)=O)=O)CCC(CC1)C(C)O2 C(CC(=O)N1CC(F)(C(N2CC(n3cnnc3)C2)=O)C1)(c1cccs1)NC(N)=O C1(NC(C2(C)CCCO2)=O)CC2CCC(C1)N2C(c1cnc2cc[nH]c2c1)=O CC1OC2(C(=O)NCCCNC(c3csc(S)n3)=O)CCC1CC2 CCC(C)(C(=O)NC1CCN(C(=O)CC2(C)CCC2)CC1)C(F)F N1(C(c2n[nH]c(C)c2O)=O)Cc2n[nH]cc2C1C(=O)NC1CCn2ncnc2C1 C1(C)(NC(C(C)N(CCC)C(C2(COC)CC=CC2)=O)=O)CCCCC1C c1(C(N2CC(NC(CC(CC)C3CCC3)=O)C2)=O)ccc(C(F)F)c(C)c1 c1(C(=O)NCC2(F)CN(C(C(CC)OCC)=O)C2)ccc(F)c2occc12 C12(C(=O)NC(C)CC3CCC3)CCC(CN(C(C3(C)CC3(F)F)=O)C1)C2 c1(OC)ccc(O)c(C(=O)NCC2CN(C(c3cscc3Cl)=O)CCC2C)c1 N1(C(CC(CNC(c2ccccn2)=O)OC)=O)CC2(CCC1C1CC1)CC2 C(=O)(C1SCCc2ccccc21)N1CCC(O)(CNC(CCCCCOC)=O)C1 CCC(CNC(=O)Cn1cc(C2CC2)nn1)(CC)NC(=O)CN1CC(C)(OC)C1 c1(C(=O)NC2CC3(C(NC(c4c(C)nns4)=O)C3)C2)cc2nccnc2cc1C c1(C(=O)NCC(N(C(CC2C(C)C2)=O)C)C2CC2)c(O)ccc(Cl)c1O C(CC(=O)N(CCCN=[N+]=[N-])C)(C(C)C)NC(C(CCC)C)=O C1(C(F)F)(CNC(CSCCOC)=O)CCN(C(=O)Cc2nc[nH]n2)C1 N1(C(c2c(C)scc2)=O)CCC2(CC2NC(=O)Cn2ncn(C)c2=O)C1 C1(C(=O)NC2CC(CC)C2)CC=CCC1NC(c1cnnn1C)=O c1(CNC(Cc2cc(CC)no2)=O)ccccc1F.C12CC(C1)CC(=O)N2 c1(NCc2n(C)ncc2)ncc(-c2cccnc2NC(=O)OCC(F)(F)F)cn1 Cc1csc(C(N2CCC(NC(c3ccoc3)=O)CC2)=O)c1Br c1(CC(C)C)cc(C(=O)NCC(C2CC(C)(C)CO2)O)c(C(C)(C)C)[nH]1 c1(NC(C2CCN2C(c2ccncc2O)=O)=O)ccc2c[nH]nc2c1 c1(OC)ccc2ncnc(NCC3(NC(c4ccc[nH]4)=O)COC3)c2n1 N1(C(=O)COCC(F)F)CC(CO)C2(CCN(C(c3c[nH]c(=O)cn3)=O)CC2)C1 C(=O)(C(C)(CSC)NC(C1C2CCCCC12)=O)NC1(CCOC)CC1 C(=O)(C(O)C1=CCCCC1)NC(CCOCC)C(N1CC2(CCOCC2)C1)=O c1(C(=O)NC(CC)(CNC(=O)C2=NOCC2)CC)cc(C#N)cc2ccccc12 N1(C(c2c(CC)nns2)=O)CCOCC(CNC(c2cccc(O)n2)=O)C1 C1(CCNC(=O)CC2(NC(C3CN4CCC3C4)=O)CC2)CCCCC1O C(=O)(C(C)S(C)(=O)=O)NCC(CC=C)NC(=O)C(C)(C)C(F)F Cc1ccc(CCNC(C2(N(C)C(c3ocnc3C)=O)CC2)=O)nc1 c1(NC(C23CC(NC(c4cc(C)no4)=O)(C2)C3)=O)ccc(Br)nc1C C1(N(C(C2(C(=O)Nc3n(C(CC)C)ncc3)CC2)=O)CC)CCN(CC)CC1 c1(CCC(N2C(CNC(=O)CC3CC=CC3)CC2)=O)cc(F)cc(Br)c1 c1(C(C(=O)N(CCNC(=O)C(C)(CO)NC(C)=O)CC)C)ccc(F)c(F)c1 C[Si]1(C)CCCCN(C(=O)CCC(c2cc(Cl)ccc2Cl)=O)C1 CC(CN(C)C)C(=O)N1CCC1CNC(C1CCC(c2ccccc2)O1)=O Cn1cnc2cc(C(=O)NCC3CC(O)CN3C(=O)Cc3cc[nH]n3)ncc12 C#Cc1cccc(CN2C(C(=O)NC3(c4cccc(Cl)c4)CC3)CC2)c1 C12(C(=O)NCOC(C)(C)C)C3C4C1C1C2C3C41C.C1(OC(C)C)CC2N(C1)C2=O C(=O)(C(C)(C)NC(C)=O)NCCN(C(CC=CCC)=O)C1CCOC1 C1(C(N(CC#N)CC2CCCOCC2)=O)C2CC(F)(F)CC12 c1(C(N2CC(C(C)NC(c3ccn(CCC)n3)=O)C2)=O)coc2c1COC2 c1(CC)ccc(O)c(NC(c2c(CNC(=O)C=CC3CCOC3)nnn2C)=O)c1 c1(NC(CC2C(CNC(CCC)=O)C2)=O)cccc(N2C(=O)CCC2=O)c1 n1(Cc2c(C)cc(I)cc2)cnnc1S(=O)(=O)C(C)(C)C C1(C(=O)NC2(CNC(CC(C)c3cnn(C)c3)=O)CCC2)CC2C=CC1O2 C1(O)(CNC(c2cn(C(F)F)cn2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C1 CC(CNC)C(=O)NOC(C12CC(CO1)C2)C.c1(C)cncn1C c1(OC)nc(=NC2CC(F)(CNC(=O)C(F)(F)C3CC3)C2)nc(OC)[nH]1 c1(C(C(=O)OC)OCCOCCOCC)ccn(C)c(=O)c1.C1(CC)C(=O)N1 N1(C(c2c(OC)cnc(-c3cnc(N(C)C)cc3C)n2)=O)CCN2CCC1CC2 C(=O)(C(F)(CC)C(=O)OC)NCC(C1CCC1)NC(c1cnc(CC)nc1O)=O c12cc(cc(F)c1)C(=O)NOCc1cn-2nn1.C1(C(C)(C)C)CC(=O)NC1=O C(=O)(C1=NN(C)C(=O)CC1)NC1C(NC(CC(CC)CN(C)C)=O)CCOC1 CCC(O)C(C)C(=O)NC(C)CC1CCN(C(C2(c3ccccc3F)CC2)=O)CC1 C1CC2=CCN(CC2)C(=O)C(C)=NO1.C=C(C)CCC(=O)NC(C)C CC1CC(C(=O)NCC(C)CC(=O)NCCC(Cl)Cl)CC(=O)N1 C12(C(N3CC(C(C(=O)NC(CC#C)CC)OC)C3)=O)CCC(C1)OC2C C1(CC(N)=O)(NC(Cc2c(C)occ2)=O)CCN(C(C2CCC2C(N)=O)=O)CC1 Cc1cccc(N)c1C(=O)NC1CCCC(N(C(=O)CCN2CCOCC2)C)C1 Cc1sc(=O)n(CCC(=O)NCC2CN(C(C3(C#N)CCOC3)=O)CCO2)c1C CCCC(C(=O)NC(C)(CNC(c1ccc(C(=O)OC)nc1)=O)C(C)C)N(C)C C1(CNC(C2=CN(C3CCC3)CC2)=O)CC2(CCC2)CN1C(=O)C(O)C1CC1 Cc1cc(C(=O)OCC2CC2)nc(CO)n1.c12ccc(C)c(c1)O2 N1(C(C2CC(=O)NC2)=O)CC2CCN(C(=O)Cc3ccc(Br)nc3)C2C1 c1(N2C(NC(CC)Oc3ccccc3)CCCC2)cc(C)nc(C)n1 c1(N(C)Cc2n(CC)cnn2)ncnc(NCCC2CCCN(C)C2)c1C N1(Cc2c(C)n[nH]c2)CCC(O)(CC(=O)Nc2ncccc2I)CC1 c1(CC)csc(S(=O)(=O)NC(=O)NCCc2cncn2C)n1 N1(C(=O)NCc2ncn(CC)c2)CCCC(c2ncc[nH]2)C1 c1(CC(N2CCC(NC(c3cnn(CCOCCO)c3)=O)C2)=O)ncn2c1CCC2 c1(C(=O)NCCN(C(=O)C(C)(C)C(F)F)C)cnn2c1OCC(O)C2 c1(OCC(N2CC(C(F)(F)F)C2)=O)cccc(CNc2cnc(C(F)(F)F)cn2)c1 C(CCCCCC(N1CCC(O)C1)=O)NC(c1cn(CC=C)nc1)=O C1(C(N2CCCN(C(c3ccc(N(C)C)nc3)=O)CC2)=O)CCN2CCCC2C1 C(C(C)CC(=O)NCCc1ccncc1)NC(Cn1ccc(C)n1)=O CC(C)(O)C(F)C(=O)NCC(C)(C)NC(=O)C(O)Cc1cnc[nH]1 C12(NC(c3cncc(OCC(F)F)c3)=O)CC3CCC(C1C2)N3C(=O)CC(F)F c1(OCC(=O)NCC(C)NC(C=CSC)=O)cccc(C(C)(C)C)c1 C1(CS(N)(=O)=O)CN(C(=O)CCc2cnc(O)[nH]2)CCO1 CCCCN=C(NCC1CCCCN(C)C1)N1CCC2(C1)CC(F)(F)C2 C1(C(=O)NCC2(C)C(C)CN(C(=O)CNC(=O)C3CC3)C2)CCn2cnnc2C1 C1(OC)COCC1NC(C1CCOC1CNC(=O)CC1(CN(C)C)CCCC1)=O c1(C(C(N2CCC(N(C(c3ncc(C(=O)OC)s3)=O)CC)C2)=O)C)c(C)n[nH]c1C Cc1ccc2nc(SCC(N3CCN(C(C4CSCCS4)=O)C(C)C3)=O)[nH]c2c1 N1(C(Cc2n(C(C)C)cnn2)=O)CC(O)CC1C(=O)NCc1[nH]nnc1C Cc1cccc2[nH]cc(C(=O)NCC3(NC(c4csc(C#N)c4)=O)CCCC3)c12 C1(C(=O)NCC(CNC(c2cnn(C(C)C)c2Cl)=O)C)CCC(C)(C)CO1 Cc1ccc2[nH]nc(C(=O)NCCOCCN(C(=O)C#CC3(C)CC3)C)c2c1 C1(OC)CC(CO)N(C(C2CCN(C(=O)Cc3c(C)noc3Cl)C2)=O)C1 C1(C(=O)NC(C2N(C(c3c(C)[nH]cc3)=O)CCC2)C)CCCN1N=O CC1CN(C(=O)NC2CCC2c2ccccc2Cl)CCc2ccc(O)cc21 C=CC1(CC(=O)NCc2ccnn2C(C)C)CCC1.C1(C)C=CC(=O)NC1 c1(NC(C(N2CC3(C(C(=O)OC)C3)C2)C2CC23CCOC3)=O)c(C)cccc1C c1(CCCC(=O)NCC(C)CNC(C2(O)CCC2)=O)nc2ccccc2[nH]1 CC1CN(C(=O)Cc2ccoc2)CC(C)CN1C(=O)CCc1ccon1 C12(CC(=O)N(CCC)CCNC(=O)COC(C)C)CCC(C)(C1)OC2 CCC(C)(C)CC(=O)NC(C)CCNC(=O)C1=NOC(C(C)(C)C)C1 N1(C(C2CC(OC)C2)=O)CCC(C(C)(C)NC(c2ccnn2CC(C)C)=O)C1 Cc1ccc(F)cc1S(=O)(=O)N1CCN(c2ncnc3c(Br)c[nH]c23)CC1CO CCCC(CC)C(=O)NC1CC(C)N(C(=O)C=Cc2cccc(Cl)c2)C1 c1(C(=O)NCCN(C(C=CC)=O)CC2CCCCC2)c(C(F)(F)F)nc(C)n1O c1(C(=O)NC2C(CNC(CC(CC)C)=O)CCC2)cc(C)c2sccc2c1 C1(C(N(CC(CC)OC)C)=O)CCC(C)(C)N(C(c2cc(C)n(C)n2)=O)C1 c1(C(c2nnnn2CC)NCCC(CCC)C)cc(C2CC2)ccc1Br CCCCCC(CCC)(c1nnnn1CC)NCCCOc1ccc(F)c(Cl)c1 C1(NC(C(C(C)C)NC(C)=O)=O)COCCN(C(C2(C#N)CCCCC2)=O)C1 Cc1cc(C(=O)NC(C)(C)CNC(=O)C(C)N(C)C)c(N)c(Cl)n1 C1(OC)(CNC(c2nc(C(C)C)oc2C)=O)CCN(C(C2COCC2(C)C)=O)C1 C1(CC(=O)NC(C(=O)N(C)CC)C)CCCC(NC(=O)C=C2CCC2)C1 CC1(C)CCC(O)(CNC(=O)CCCCN(C)c2cc(C(N)=O)ncn2)C1 c1(C(N2CC(CNC(CCOc3ccc(C)cc3)=O)C2)=O)c(F)cc(Cl)cc1F Cc1ccc(C(N2CC(N3CCCC3=O)C2)=O)cc1C.C12CC(C)(C)CN1C2=O c1(C(=O)NC(C(C)C)C(C)NC(=O)CN(C2CCC2)C)cc(N)c(F)cn1 C1(NC(c2nccs2)=O)CN(C(=O)Cc2cnccc2Cl)Cc2nccn2C1 S1(=O)(=O)c2cccc(c2)N1.CCCCCCN(C)C(=O)NC(C(N)=O)C(C)C N1(C(C2CCSC2)=O)CCCC(n2cc(CNC(c3cccc(O)c3)=O)nn2)C1 N1(C(C2C3(CCN(C(C(=C)C(F)(F)F)=O)C3)C2)=O)CCC2(CC1)COC(C)C2 C1(C2(C(=O)NCc3cnc(O)s3)CC2)CCCN1Cc1coc(C(F)(F)F)c1 C1(NC(C(C)N(C(=O)C(C)C(=O)OC(C)(C)C)C2CC2)=O)(CO)CCCCC1 N1(C(C2OCC(C)(C)C2)=O)CCN(C(C2(Br)CC2)=O)C2(CCC2)C1 n1(Cc2nc(C(C(C)C)C)nn2-c2ccnn2C)nc2n(c1=O)CCOC2 C(=O)(C(C)(C)CC(C)(C)C)NCC(C1CC1)NC(COc1c(C)c(Cl)ccc1)=O c1(CC)ccc(C(=O)NCC(C)(Cn2cccn2)NC(=O)CC(C)c2ccco2)o1 C1(C(N2CC3CN(C(C(C)C(C)(C)C)=O)CC3C2)=O)CCC2CC(C)CN2C1 C1(C)(CNC(C2C(C)CN2C(=O)CCc2cccnc2)=O)CC=CCC1 C12(CNC(C(C(C)(C)C)O)=O)CN(C(c3cccc[n+]3[O-])=O)CC1CCO2 N1(CC(=O)NC2(CNC(C3CCC3)=O)C(C)CCCC2)CCc2ccccc21 C(=O)(C(F)(F)Cc1ccc(F)cc1)NCC(C)(C)N(C(C(C)C1CC1)=O)C N1(C(=O)CCC2CCC2)CCC2(CC1)CCN2C(c1cc(Cl)sc1Cl)=O N1(C(N(C)CC)=O)Cc2ccccc2CC1CCc1nn[nH]n1 C1(NC(c2nc(C(C)OC)sc2)=O)CCCN(C(=O)C2CC2)CCC1 N1(C(CCN(C)C)=O)CCC2(CC1)CC2C(=O)N(CCC#N)Cc1ccccc1 N1(C(C2=C(C)CCC2)=O)CCCC12CCCN(C(=O)C1=CS(=O)CCC1)C2 CS(=O)(=O)C1CCCN(C(C2CCCN2C(=O)CC2CCC2)=O)C1 Cc1nn(C)c(Cl)c1C=CC(=O)NC1CC(CNC(=O)CCC(C)C)C1 c1(NC(CC)C2CCC2)ccc(N2CCN(CC)CC2)cc1 C1(C(=O)NC2C(NC(c3c(CC)non3)=O)COC2)Cc2cc(F)cc(F)c2O1 C1(CCCNC(C2N(CC)CC2)=O)CCN(C(=O)CC2COCCN2CC)CC1 CN1CCCC(NC(C2N(C(c3cccc(Cl)c3)=O)CC2(C)C)=O)C1=O O=C(CC1=CCOCC1)NC1C=CCN(c2nnc(C(F)F)s2)C1 C1(CC)CN(C(c2cn(C3CCC3)nn2)=O)CCN1C(=O)C(c1cccnc1)C C1(c2n(-c3c(C)cc(C)cc3C)nc(-c3nccs3)n2)CCc2nnn(C)c2C1 c1(C(C)C)ccccc1CC(=O)NCCC(C)NC(=O)CN1CSCCSC1 c1(C(N2CCC(N3CCNCC3)C2)C)cc(Br)ccc1O c1(CC(=O)N)ccc(OC)cc1.C(CCNC)N(C(=O)C=CC(=O)OC(C)C)CC C1(NC(CSCCOC)=O)CN(C(=O)COc2ccccc2)CC(C)(C)O1 C1(CC=C)(NC(=O)CC2CC(F)C2)CCCN(C(=O)Cc2ccc(C)cc2C)C1 Cn1c(=O)n(C)c2cc(C)ccc12.N1(C(C2CC2(F)F)=O)C2CCC1CC(N)C2 c1(CC(N2C(C(=O)NCc3c(OCC=C)cccn3)CC2)=O)ccc(O)c(Cl)c1 C1(NC(COC)=O)CC(C(F)C(=O)NC(CCO)C2CCC2)C1 C1(CNC(c2n(CC)cnn2)=O)CCC(C)CN1C(C12CC(CC(F)F)(C1)C2)=O c1(C(=O)NCC(C)N(C)C(c2ncn3ccccc23)=O)c(N)cc(Cl)cc1F c1(C(N2C(C(=O)NCC(C)(F)F)CC(F)(F)C2)=O)cccc([N+](=O)[O-])c1I C(=O)(CCCC(=O)NC)N(C1C(NC(c2c(CC)nc[nH]2)=O)CCCC1)C c1(C(=O)NC2C=CC(CNC(C3CC(O)C3)=O)C2)nnn2ccccc12 c1(OCCC(=O)N(C2CCN(C(=O)C(N)=O)C2)CCC)ccc(C)cc1C N1(C(C2(S(C)(=O)=O)CCC2)=O)CCC(C2(NC(=O)CC3CNC(=O)C3)CC2)C1 N1(C2C(=O)N2)CCC(OC(F)F)C1.C#CCCN(C(=O)CO)C c1(C(=O)NCC(CNC(CC2CC(OC)C2)=O)C)cc2c(ccn2C)[nH]1 c1(C(C)C(N2CC(C)(CC(N3CCCCC3CO)=O)C2)=O)ccc(F)cc1 N1(C(c2ccc(C#C)cc2)=O)CCC2CN(C(c3ccc(F)nc3C)=O)CCC12 c1(CC(N2C(CN(C(c3c(OC)scc3)=O)CC)CCC2)=O)cn2cc(C)sc2n1 c1(C(=O)NC2C(CNC(C3C(C=C)CC3)=O)COC2)ccccc1C(C)=O Cc1cnc(N(C)CCc2csc(C)n2)c(S(=O)(=O)N2CCCC(F)(CO)C2)c1 O=C(N=S(=O)(CC1(c2ccccc2)CC1)c1cccc(Br)c1)c1ccc(Br)cc1 CCCCC(CC)CCC(COC(C1(C)CCN1C(C)=O)=O)CC C(=O)(C(F)(F)CCn1ccnn1)N1CC(NC(C2CC2[N+](=O)[O-])=O)C1 N1(C(c2cc(CC)sn2)=O)Cc2occ(C(=O)NCC3CCCNC3=O)c2C1 C1(NC(C2(OC)CCOC2)=O)CC2(C(=O)NCC(C)CC(C)C)COC1C2 CC1OC2(C(=O)NC3CCCN(C(c4sccc4C(C)(C)C)=O)C3)CC1C2 c1(CC)nn(C)c(CC(N2CC(NC(C3CCC(=O)N3)=O)C(C)C2)=O)c1Br C1(O)(C(c2ccccc2F)C)CCN(C(=O)CN2C(=O)CCC2=O)CC1 c1(C(=O)NC2C(CNC(c3c(C)cc(C#N)cc3)=O)C2)ccc2c(c1)COCC2 c1(CNC(C(=O)NCC(C)(COC)OC)=O)ccc(CCN)cc1 N1(C(COCC(C)(C)C)=O)CC2CCC1CN2C(C1CCCCS1)=O C1(C(=O)NCC2(OCC)CN(C(=O)Cc3sccc3C)C2)CC2CCC1CC2 C1(=O)C(C)C(=O)N2CCOCC2C(=O)CO1.N1(CC)CCCCC1C S(=O)(=O)(c1ccccc1[N+](=O)[O-])Nc1ccc(OCCCC)nc1C C1(CC(=O)NC(COC)CCO)CN(C(=O)COC(C)=O)C(C)(C)C1 O=C(COc1cccc(I)c1)NNC(=O)C1NC2CCC1C2 C1(CCNC(COCC#C)=O)CN(C(=O)C(F)(F)CCn2ccnn2)CC(C)O1 c1(C(N2CC(F)(C(N3CCOC4CC34)=O)C2)=O)cccc(I)c1F C1(Cl)(C(N(C2CN(C(c3cc(OC)no3)=O)C2)C)=O)CC12CCOCC2 Cc1coc(C)c1C=CC(=O)NC1(CNC(C23C=CC(CC2)C3)=O)CCOC1 CCCC(O)(CCC)CC(=O)NCC=CC(=O)NCC1CNC(=O)CO1 Cc1ccc(=NCCC(=O)NC2CCCC23CCN(C(=O)C2=CCC2)CC3)[nH]c1 N1(C(c2ncc(OC)nc2)=O)CC2CC(CNC(=O)CCOC3COC3)CC1C2 c1(OC)cccc(OC)c1C(=O)NCC1(NC(=O)C(C)P(C)(C)=O)CCOCC1 C(C(C)(C)C(=O)NCC(=O)NCC(=O)Nc1cnncc1OC)SC C1(CC)CCOCCN1C(=O)C(N1CCC(COC2CCOCC2)CC1)=O C1(OCC)CC2CCC(C1)N2Cc1cn(C2CCCCC2)nn1 N1(C(c2cc(-c3ccc(OC)cc3)no2)=O)CC2C3CCC(C3)C2(C)C1 c1(C(=O)OC)ccc(NC(=O)N(C)CCc2nc(=O)o[nH]2)cc1OC c1(C(N2CC3C(CN(C(=O)C(F)OC(F)(F)F)C)C3C2)=O)nnn2ccccc12 c1(C(=O)NC2CCCCC2NC(c2c[nH]nc2Br)=O)ccc2c(c1)CC2 c1(C(=O)NCC(CC(=O)NCCCOCC)OC)cc(C)c2n[nH]cc2c1 c1(-c2cccc(C#N)c2)nc(C2SCCc3ccccc32)n(C2CCSCC2)n1 C1(O)(CNC(CN(C(C=CC(C)(C)SC)=O)C)=O)CCN(C)C1 O(N=C1CCCCCC1)CC(=O)N(C1CN(C(c2cc(CC)nn2C)=O)C1)C C1(NCC2CC(NC(c3ncn(C)n3)=O)C2n2cccn2)CCC(F)(F)C1 N1(C(Cc2ncc(C)[nH]2)=O)CCCN(C(=O)CCn2nc(C)nc2C)CC1C C1(NC(C=Cc2ncc(C)[nH]2)=O)(CO)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 C1(CC=C)(NC(=O)C(O)c2ccco2)CN(C(C2CCC=CO2)=O)C1 c1(C(N2CC(C(C)NC(c3coc(Cl)c3)=O)C2)=O)cc(F)cc(Cl)c1 N1(C(C(c2cccnc2)C)=O)CCC2(CCCN(C(C3(N(C)C)CC3)=O)C2)C1 c1(N(C(C)CNC(=O)Cc2cnc[nH]2)C)nc(Cl)ncc1C1CC1 C1(C(=O)NC(C)(CNC(c2c[nH]nc2[N+](=O)[O-])=O)C2CC2)CCC(=C(F)F)CC1 CC1(C#CC(=O)N2CCCC(NC(=O)C(c3cccc(Br)c3)O)C2)CC1 c1(C(=O)NCC2CCN(C(c3n(CC)ncc3Cl)=O)CC2)c(C)nc(C)nc1C Cc1cc(C(=O)NCCCCN(C(=O)Cc2csc(C3CC3)n2)C)cc(F)c1C c1(CNC(=O)Nc2cc(C(=O)OC)ncc2)c(C)n(C)c2ccccc12 c1(SC2CC(NC(=O)C=C(Cl)Cl)C2)ccccc1.CC1C(=O)NCC=CC(=O)O1 c1(OC)cc(Cl)c(NC(C2(C)CCN(C(c3cccc(F)c3Cl)=O)C2)=O)c(Cl)c1 C1(NC(CC(CC)C(F)F)=O)CCN(C(=O)CC(C)(C)OC)CCC1(F)F S(=O)(=O)(c1cnc(Cl)cc1Br)N(C1CCOC1)C Cc1cc(=NC(=O)C2CC(NC(=O)C(O)CN(C)C)C2(C)C)[nH]n1C C=CCC(C(=O)N1CC(NC(=O)OC(C)(C)C)C1(C)C)C(C)C C1(C(=O)OC(C)C(=O)NCCS(=O)(=O)c2ccccc2)CCCN2CCCCC12 c1(C(=O)NCC(CN(C(C(C)=Cn2ccnn2)=O)C)C)cc2cc(Cl)ccn2n1 c1(-c2nc(N3CCN(C(C)=O)CC3)nn2C2CCOC2)cc(F)ccc1C CC1COCCN(C(=O)C(c2cccs2)NC(c2ncc[nH]2)=O)C1 CC1CN2CCN1CC2C(=O)NC1CCC1NC(C1CCS(=O)(=O)C1(C)C)=O CC1(C)C2CCC(C2)C1NC(C1CCC(NC(c2cc(Br)c[nH]2)=O)CC1)=O C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1CC(N(C(C2N3CC(C)N(CC3)C2)=O)C)C1 CC1(C(=O)NCC2(CNC(c3ccc(=N)[nH]c3)=O)CC23CCC3)COCCO1 C(=O)(C1=CC2(CCOCC2)C1)N(C1CCN(C(C2CC2C(F)F)=O)CC1)C c1(C(N2C(C(N3CC(CN(C)C)OCC3)=O)C=CC2)=O)ccc2nccnc2c1 CS(=O)(=O)CCc1cn(CC2CCN(C(=O)C=CCOC3CCCCC3)C2)nn1 C1(C)(CC)CC(NC(=O)CCC(=C)Br)CN1C(C1CCOCC1)=O N1(C(C(C(CC)O)(C)C)=O)CCc2nc(CNC(c3cc(Cl)cn3C)=O)sc2C1 c1(C(=O)NC(c2cccnc2)CNC(C2(CSC)CC2)=O)cc(N)cc(F)c1 c1(C(CC(=O)OCC)NCCC(C2CCOCC2)C)ccc(F)cc1 CC1CCN(CCc2cnc(C(=O)N(C)C)nc2)CCN1 CCC(CC(=O)N(CCCN(C)C(C1C2CCC1(C)C2(C)C)=O)C)C(C)(C)C C1(C(C)=O)C2CC3C(C2=O)C13.c12ccc(c(F)c1)o2.C1(C)C(=O)O1 C1(C(C)NC(C=C(C)C2CC2)=O)CCCN(C(=O)Cn2cnnc2)C1 C1(CNC(C2CC(C)=C(C)CC2)=O)CC2(CO1)CN(C(=O)C(C)N(C)C)C2 C1(C(N(CC(C)OC)C)=O)(CNC(C2CCCS2)=O)CC(C)(C)C1 C1(C(N(c2nnc(CC(C)C)s2)C)=O)CC(C)C(C(=O)OC)O1 CCCC(CC)C(=O)NCC12CC(CNC(=O)CC(C)CN(C)C)(C1)C2 C(=O)(C(C)CO)NC(C)CN(C(=O)C(=O)NCc1ccccc1)C C(=O)(C1OCCc2ccccc21)NC1C=CCN(C(C(CC=CC)CC)=O)C1 C1(NC(=O)NCC(c2ccc(Br)cn2)C)CCCOC12CCC2 c1(C(C)NC2CN(C(=O)OC(C)(C)C)CC2C)cccc(Br)c1 C1(C2CCN(C(C3CC3C)=O)C2)(NC(C(c2c(OC)cccc2)OC)=O)CC1 C(=O)(C1=NN(C)C(=O)CC1)N1C2CC(OC(C)C)(C2)C1 C(C1CCS(=O)(=O)c2ccccc21)CNC(N1C(CC(C)O)CCCC1)=O C1(C(=O)NCC(n2cncn2)C)CC(F)(F)CN1C(C1CC1(F)Cl)=O CCC(CNC(c1sncc1C)=O)(CC)C(=O)NC1CC2CCCCN2C1 N1(C(C23COCC(C)(C2)C3)=O)CCC2(CC1)CN(C(=O)CNC=O)CC2CO C1(C(N(CCCNC(C2(c3cccc(Cl)c3)CCC2)=O)CC)=O)CC2C=CC1C2 c1(C2(CN(c3nnc(C(C)(C)C)o3)C)CCC2)ccc(OC2CCCC2)cc1 N#Cc1ccnc(COc2cccc(-c3nnco3)c2)c1 C#Cc1cccc(-c2nc(C(=O)OCCn3nc(C)c(Br)c3C)nn2CC)c1C C(=O)(CC(C)NC(=O)C(C1CCCC1)NC(C1COCC1C(N)=O)=O)OC C1(C(=O)NC2CC(CNC(C(CC)N3CCCC3=O)=O)C2)C(C)OC(C)C1C c1(C(N2CCC(N3CCCC3)C2)C(=O)NN(C2CC2)CCF)cc(Cl)c(Br)cn1 c1(-c2nc(C(C)(C)C)on2)ccc(OC(c2ccc(NS(N)(=O)=O)cn2)=O)cc1 C=C(C)CC(C(=O)N1CCCCC(N(C)C(c2ccncn2)=O)C1)OC N1(C(C(C(CC)O)C)=O)CC2CCC(NC(C3CN4CCN3CC4)=O)CC2C1 C(CCCC(=O)N1CCC(O)(CNC(=O)CC2CCCN2C(C)C)C1)OC C1(CNC(c2c(OC)cccn2)=O)CN(C(=O)Cc2cc(C)[nH]n2)CC12CCC2 c1(C(N2CC(NC(c3cccc(CC)n3)=O)C3C2C3)=O)ccc(C)cc1O c1(NC(C(=O)NC(C2CCOCC2)CC)=O)ccnn1-c1cnccn1 C1(CC(=O)NC(c2cn[nH]c2)C)CCCCC1NC(=O)Cc1cnn(C)c1 c1(C(=O)NC2CC(NC(C3C(=C)C3)=O)C2)ccc(=O)n(CCCC(F)(F)F)n1 c1(SC(C)C(=O)NC2CCC(NC(c3ccn(C)c3)=O)C2)ccc(F)cc1 c1(C(N2CC(NC(C34CCOC3CCOC4)=O)C2)=O)cc(Br)cc(F)c1F Cc1nc2c([nH]1)C(C(=O)N1CCC3C(C1)CN3C(=O)COCC(F)F)CCC2 C(C(C)CC(=O)NC1CCCC1(C)NC(c1cc(C)n(C)n1)=O)OC N1(C(C(CC=C)C)=O)CCCC2(CCCN2C(=O)C(C2CCCCCCC2)O)C1 CCC(C)(CNC(C1CN(C(C)C)C1)=O)C(=O)NCC(C)C(=O)OC c1(N2CCN(C)C(CNC(=O)CN3CCCC3)C2)nc(O)n(C)c(=O)c1[N+](=O)[O-] c1(CC(=O)NCCCNC(C2(F)C(C)OCC2)=O)c(Cl)cccc1Br Cc1cc(N)c(C(N2CC(CNC(=O)CCCN3CCCC3)CC2C)=O)cc1C c1(NC)nc(C)ccc1C(N1CCN(C(C2C3CC4C(C3)C24)=O)CC1)=O c1(C(=O)NC(C)CCCCNC(C2CCCO2)=O)cc(Br)c(F)cc1F N1(CCNC(=O)OC(C)(C)C)CCCN(C(C2(C#N)CC2C(F)(F)F)=O)CC1 C=CCC(CC(=O)N1CC2CC2(C(=O)OC)C1)NC(c1nn[nH]n1)=O N1(C(c2cc(N)c(O)c(F)c2)=O)CCC2(CC1)CN(C(C1CC3C=CC1C3)=O)C2 N1(C(c2n[nH]c(CC)c2Cl)=O)CCOC2(CCN(C(C3(S(N)(=O)=O)CC3)=O)C2)C1 Cn1ccc2cc(C(N3CCOC4CN(C(c5cc[nH]c5)=O)CC34)=O)ccc12 C(=O)(C1=C(C)CCC1)N1CC(SC)C(NC(C2(C(C)C)CC2)=O)C1 C(=O)(C(C(=O)NCC(C)CNC(=O)C=C(C)c1cnn(C)c1)C(C)C)OCC CC1CCOC(C(=O)NC(C)C(C)NC(=O)CCc2nc(O)n[nH]2)C1 c1(CN2CC(C(=O)NCc3ncc(Br)s3)C(O)CC2)c(F)ccc(Br)c1F C1(NC(c2cc(C)c(C)s2)=O)CCC2CCN(C(=O)CC3COC(=O)C3)C1C2 C1(O)(CCC(C)(C)NC(=O)CC2CCCCC23CC3)CCCN(C(=O)C(N)=O)C1 C1(NC(C2OCCN(C)C2)=O)CN(C(=O)Cc2ccc(F)cn2)CCC1F C(C(O)CC(=O)N(C)CC1(O)CN(C(=O)CCc2cccc(O)n2)C1)N(C)C C=CC(CCC)CC(=O)N1CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC(C)C1 c1(CNc2scc(-c3ccc(C(=O)NC(C)C)nc3)n2)c(Br)cc(F)cc1Br c1(CC)nc(C)ncc1C(=O)NC1CCCCC1NC(C1CC(C)CCO1)=O N1(C(C2N(C)C(=O)NC2)=O)CC2CCC1(CNC(=O)Cc1cnccc1Cl)C2 C1(CNC(=O)Cc2ccco2)CC(NC(c2csc(F)c2)=O)C12CCC2 CC12CN(C(c3ccc(Cl)o3)=O)CC1CN(C(c1cc(=O)c(OC)co1)=O)C2 C(=O)(C(C)S(C)(=O)=O)N1CCC(CCNC(c2c(Cl)cn(CCC)n2)=O)CC1 N1(C(CNC(CCOC(C)=O)=O)=O)CC(C(=O)NOC(C)CC(C)C)CC1(C)C CN1CCCC(NC(=O)C(CC2CC2)NC(c2ccnc(CO)c2)=O)C1 N1(C(CNC(C(C)CC2CC2)=O)=O)CCN(C(=O)C=Cc2ccsc2)CC1 C(=O)(C1=CC2(CCN(C(C)=O)C2)C1)N1C(C)CC(C(=O)OC)CC1C c1(CC)nn[nH]c1C(=O)NC(c1nocc1C(=O)NC1(CCO)CCOC1)C C(C(=O)NCc1ccc(F)c(CO)c1)(C(C)(C)C)SC O=C(C(F)(F)C(F)(F)F)NC1C2CCC1CN(C(c1ccc(C3CC3)cc1)=O)C2 N1(C(c2c(CC)scc2)=O)CC2COCC(C1)C2NC(=O)CC1CCCCCC1 c1(C(=O)NCC(c2ccccc2)NC(C2C(C)C2)=O)cc(C(F)(F)F)cc(N)c1 c1(C(=O)NC2C3CN(C(C4CCCSC4)=O)CC23)cnn2ncccc12 C1(C(N2CC(CC=C)(C(=O)NCCc3ncc(C)o3)C2)=O)CCOC(CC)C1 c1(C(N(C(CC)CC(=O)NCCC2CC=CCC2)C)=O)cc(O)cc(F)c1 C1(C(C)C)C(NC(=O)CNC=O)CCN1C(=O)CNc1cnn(C)c1 N1(C(C2CCCC(C)C2)=O)CCC2CN(C(c3ccc(C(F)(F)F)[nH]3)=O)CC12 CC1CCc2cccnc2N1C(c1cccc(S(=O)(=O)NCC(=O)O)c1)=O c1(OC)cc(F)c(Br)cc1C(=O)N(CCS(=O)(=O)O)CC1CCCCO1 C1(C2CC2)(CNC(C2(C#C)CCCC2)=O)CCN(c2cc(OC)nc(CC)n2)C1 Cc1cc(C(N2CC=CC(C(=O)NCC(C)CC3CCC3)C2)=O)nn1C c1(NC(CC2OCCN(C(CCC)=O)C2)=O)cccn2nccc12 CC1CN(C(c2cc(F)n[nH]2)=O)CCN1C(=O)Cc1cccc(F)c1F Cc1cnccc1C(=O)NC1(C)CCN(C(=O)CCC(=O)c2ccc(N)cc2)C1 N1(C(=O)C=Cc2cccnc2)C(CNC(=O)C(F)(F)C(F)(F)F)CC2COCC12 CCC(C)CC(=O)NC1CCC(C(=O)NCC#CCCO)C1 N1(C(C2(CC)CCCCC2)=O)CC(NC(c2ccc(N)cc2O)=O)C(C)(C)C1 N1(C(C2(COC)CCCC2)=O)CC(C(N2CCC(C(=O)OC)C2C)=O)CC(C)(C)C1 C(=O)(CC(C)CNc1ccccc1)NC(c1cn(C)nc1Br)c1n(CC)nnn1 Cc1ccncc1C(=O)NCC1CCN1C(=O)C=CC1CCCO1 C1(c2nnnn2C2CCOC2)(Nc2cccc(COCC)c2)CCN(C)CC1 c1(C(=O)O)ccc(NCc2ccc(Cl)cc2Cl)c(SCc2nc[nH]n2)c1 C12(NC(CC(c3c(C)n[nH]c3C)C)=O)CCC(CC1NC(=O)C1=CCCOC1)C2 CC(C(=O)N(C1CCN(C(C2CCN2S(C)(=O)=O)=O)C1)C)C(C)(C)O N1(C(c2c(C)onc2O)=O)CCCC(CNC(C2CC(O)C2)=O)CC1 C1(NC(c2ccc(C)cc2)=O)CC(F)(F)CC1NC(c1ccc(N(C)C)cc1)=O N1(C(c2c(C)cncc2)=O)CC2CC1CN2C(c1cc(C2CCC2)[nH]n1)=O N1(C(C2C(C)=CCS2)=O)CCOC(C(N2CCC(O)(c3cnn[nH]3)C2)=O)C1 c1(OC)ccc(CC(=O)NCC2CCCCC2NC(c2scnc2Cl)=O)c(C)c1 N#Cc1cn(C2CCS(=O)(=O)C2)[nH]c1=NC(=O)N1CCC2(CCCC2)CC1 C1(CC=C)(C(=O)N(CCCCOC)C)CCCN1C(=O)C(C)N=[N+]=[N-] C1(O)(C(=O)NCCC(C)N(CCC)C)CCN(C(=O)CCC(F)F)C1 N1(C(C(CCC)OC)=O)CCOC2(C1)CN(C(C1CCc3nnc(O)n3C1)=O)C2 C(C)(C1OCCc2sccc21)NC1C(O)CCN(c2nc(C)nc3c2c[nH]n3)C1 C1(NC(C(c2ccnn2C)NC(C2N(CC)CCC2)=O)=O)CCCCC1(F)F C1(C(C(C)C)NC(C2(CCC)CCC2)=O)CCN(C(=O)CC2(C)CC2)CC1 c1(C(=O)OCC2(C)N(C(=O)OC(C)(C)C)CCC2)ccc([N+](=O)[O-])cn1 c1(C(=O)NC(CC)CNC(c2c[nH]c(=NC)o2)=O)ccc2nc[nH]c2c1 C1(C(=O)NCC2(CC)CC2)(CCOC)CCN(C(=O)CCSC)CC1 C(=O)(C(C)(C)C(C)NC(c1cccc(F)c1F)=O)NC(c1ccnc(C)n1)C C(=O)(C(C(C)(C)C)N1CCNC1=O)N(CCCN(C(=O)Cc1cccnc1)CC)C Cc1nc(C(=O)NC2CC(O)(C(=O)NC3(c4cc[nH]n4)CC3)C2)cc(O)n1 N1(C(c2ncc[nH]c2=O)=O)CC(CNC(C2(c3cccnc3)CC2)=O)C(O)C1 C1(COC)(CNC(C2CCC(C)O2)=O)CN(C(=O)CCN2CCCC2)C1 c1(NC(C23CC(CC(C)O2)C3)=O)nc(NCc2cccnn2)c2ncn(C)c2n1 N1(C(C(CCC)=CCC)=O)CC(CNC(C2CCCC2N(C)C)=O)C(C)(C)C1 N1(C(C=CC(=O)OCC)=O)CCC(CNC(=O)CC2CCCCC2O)C(F)(F)C1 CCCCC(CNC(c1ccnnc1C)=O)NC(=O)Cc1ccc(C)o1 CC1CCC(N(C)C(c2occc2CNC(C2CCCN2C)=O)=O)C1 Cc1csc2c(N3CCN(C(c4cn5ccsc5n4)=O)C4CC34)ncnc12 c1(CNC(CN(C(C2C(C(=O)OC)(COC)C2)=O)C)=O)cnccc1Cl c1(C(N2C(CNC(c3n(C)nc(C4CC4)c3)=O)CC(O)C2)=O)ccc(F)cc1N c1(C(=O)NCC2(NC(C(C)CO)=O)CCCC2)sc(C#N)cc1Cl c1(CCOC)ccccc1Oc1ccc(O)cc1.C(=O)(C)NCCNC(C)C.SC N1(CCOC)CCOC(c2ccnn2C)C1.C1C(=O)N1CC1CC1 CCCC(C(=O)N(C(C)CCNC(=O)COc1ccon1)C)S(N)(=O)=O C1(NC(C2CC(O)CN2C(=O)CCc2csnn2)=O)CCN(C(N)=O)CC(O)C1 c1(C(N2CC(C(C(N3C(CC)CCC3)=O)O)C2)=O)cn(C)nc1CC C(=O)(C1CCc2ccccc21)NC(CCNC(C(C)OC1CCCC1)=O)(C)C S1(=O)(=O)C2CN(C2)c2nccc(n2)N1.S(=O)(=O)(C(F)(F)F)ONC(=O)C1CC1 S(=O)(=O)(c1ccc(C#N)c(NCc2ncc(Br)cn2)c1)NCC1(S(C)(=O)=O)CC1 C=CC(CC)CC(=O)N1CCOC(CCNC(C2CCCS2)=O)C1 N1(C(c2cc(C)nnc2)=O)CC2CCC1CC2NC(=O)C(C)C(F)(F)F N1(C(c2cncc(C=C)c2)=O)CCCC12CCN(C(c1nncn1C)=O)C2 C1(COC)CN(C(c2ccc(Cl)o2)=O)CCN1C(C1CC2(C1)CC2(F)F)=O N1(C(C(CN(CC)CC)F)=O)CC(N(C(=O)Cc2csc(S)n2)C)C2(CC2)C1 C1(N(C)C)C=CCN(N2CC(c3ccc(Cl)cc3)C3(CCCC3)C2)C1 c1(N(CCCC=C)C)nnc2n1C2.C1(CC2CC2)CCC(C)(C)C1 CC1C(C(=O)NCC2CN3CCC2CC3)CCCN1C(=O)C(C)OCC1CC1 N1(C(c2cnn(C3CCC3)c2)=O)CCC2(CC1)CN(C(C1CCC1F)=O)C2 C(=O)(C1=CCCOCC1)N(C1CCCN(C(C(c2ccc(Cl)cc2)=O)=O)C1)CCF C1(CNC(C2N(C)C(=O)NC2)=O)CCC2(CN(C(c3cnc(F)c(Cl)c3)=O)C2)O1 CC1CCCCCCN1C(=O)CC=CCC1(NC(C2CC2(Cl)Cl)=O)CCC1 C1(CC)CCCN(CC(=O)NC2C3CC2N(C(C2(CC(C)C)CCC2)=O)C3)C1 C1(NC(CSC)=O)CCCC1(C)NC(C1CC=CC(O)C1)=O c1(C(N2CCNC(C)C2)=O)cnc2c(Cl)cccn12.c1(OCC)ccc(OC)cn1 c1(OCC)ccc(C(N2CC(NC(=O)CC3CC3(Cl)Cl)C(C(F)F)C2)=O)nn1 C(=O)(CCC(C(C)C)NC(=O)CCC1CCCN1C)N1CCC(C(=O)OC)CC1 C1(CC)C(C(=O)NCC(C)(C)CNC(c2cnccc2N(C)C)=O)CCN1C c1(C(=O)NC2C(CNC(C(CC)OC)=O)C2)ccc2c(c1)CCOC2 O=C(CCC(F)(F)C(F)(F)F)N1CCCC(NC(C23CC(O)C2C3)=O)C1 C(=O)(C(C)(C)CC(C)(C)C)N(C1CCC(NC(C(C)Cn2ccnc2)=O)CC1)C c1(OC)cccc(NC(C2CCCN2C(c2ccnc(C)c2)=O)=O)c1 S(=O)(=O)(c1ccc2c(c1)CCCO2)N1CCC2(CC(C)OCC2)CC1 N1(C(c2ccn(CCC)n2)=O)CCCC(NC(=O)CCc2ncco2)C1C Cc1cc(C(N2CC(CCNC(=O)CC3CCC(=O)N3)C2)=O)c(C)n1C CCCC(C)(CCC)C(=O)NCCC1CN(C(c2nocc2C)=O)CCO1 c1(SC)ncc(C(=O)N(C)CCOCCNC(C2(F)CCC2)=O)c(O)n1 C1(O)(C(C)NC(CCNC(=O)OC)=O)CCN(C(c2ocnc2CC(C)C)=O)C1 N1(C(CCC(C)(C)F)=O)CCCC2CN(C(C3CCNC3=O)=O)CC12 c1(OC)cccc(-c2nc(C(N3CC(C)(C)C3)C3(CO)CC3)n(C3CCC3)n2)c1 C1(C(=O)NCC(CN(C(COCC(C)C)=O)C)(C)C)=NC=NNC(C2CC2)=C1 C1(NC(C2C(C)(C)COCC2)=O)CCC2CN(C(=O)CCOC3CC3)CC12 c1(CC(=O)N(CC(C)NC(C2CC(C)(C)O2)=O)C)cccc(OCC(F)(F)F)n1 c1(C(=O)NCCC(C)NC(=O)CCc2ncccn2)c(F)ccc(F)c1F c1(NC(=O)NCCCCSCCC(=O)OC(C)(C)C)ccc(N)c2cnccc12 N1(C(c2n(C)ncc2N)=O)CCN(C(=O)C(C)(C)CCCO)CC(C)(F)C1 N1(C(C2CC2(F)Cl)=O)CCN2CCN(C(c3n[nH]c4c3COC4)=O)CC2C1 N1(C(C(C(C)C)CNC(C2CCCCC(=O)C2)=O)=O)CC(=O)N(C)CC1C c1(C(N2C(C(=O)NCC=C)CC(CC)CC2)=O)cnc(C)c(C#N)c1 C(=O)(CCC(F)(F)C(F)F)N1CCCC(F)(CNC(C=CCOC)=O)C1 c1(C(N2CC(CNC(c3cc(C)n(C)n3)=O)OCC2)=O)cc(Cl)c(Cl)cc1F c1(C(=O)NCCOCCNC(C=Cc2c(C)ccs2)=O)cc(C2CC2)nnc1O C1(CNC(C(C(C)C)N(C)C)=O)CN(C(C2CCC2(F)F)=O)C2(CCC2)C1 N1(C(C(C(C)NC(=O)C(O)C2CC2)(C)C)=O)CCN2CCOCC2C1 c1(C(N2CC(NC(CC(CC)CC)=O)C3(C2)CC3)=O)ccc(F)c(C)c1C N1(C(C2CC(CC)OCC2)=O)CCN(C)CC1CNC(C1(C(F)F)CC1)=O N1(C(c2cc(C(N)=O)no2)=O)C2CCCC1CN(C(=O)CC1CCSCC1)CC2 CC1CC(C(=O)N(CCC(=O)C(N)=O)CCO)CCN1C(=O)C1=CC(C)(C)C1.OC c1(C(N2CCC(C3(NC(C(CCC)OC)=O)CC3)C2)=O)ccc2cnccc2n1 Nc1ccc(Cl)nc1C(N1CCCCC1CCCNC(=O)CC1CCOC1)=O C1(CNC(COC(CC)C)=O)CCN(C(c2ccc(C(C)C)o2)=O)CCC1(F)F c1(C(=O)NCCC2OCCN(C(CC(=C=C)C)=O)C2)cccc(C(F)(F)F)c1N C(C(C)(C)CC(=O)NC(C1CCN(C(=O)COCC(F)F)CC1)C)NC(C)=O C1(CNC(C(CC)(C)CC)=O)CCCC2(CN(C(=O)CCC3CCOC3)C2)O1 c1(C(N2CCC(CCNC(C3COC3)=O)C2)=O)ccnc2c(Br)cccc12 N1(C(CC2C(C)OCC2)=O)CCC(C2CN(C(C3CCC4CC4CC3)=O)C2)CC1 Cc1ncccc1CC(N1CCCCC1C(=O)NC(c1ccccc1)CF)=O CC1(C)CN(C(=O)Cc2ccc(O)cc2Cl)CCC1NC(=O)CCN1CCCC1 C1(C(=O)NCC(C)(C)NC(c2c(O)ncc(CC)c2)=O)CCC(=O)N2CCCC12 C1(N)CC(CO)C2CC12.c1(C(N2CCCC2CO)=O)ccc(NC(c2cncs2)=O)s1 n1(CCCNC(C2N(C(C(C)(C)OC)=O)CCC2)=O)cnc2ccsc2c1=O c1(NC(C23N(C(C(C)N(C(C)=O)C)=O)CCC2C3)=O)ccc(F)cc1CO N1(C(COC(C)C)=O)CCC(C(=O)ON(C(=O)CC2C=CCC2)C)CC1 N1(C(COCCOC)=O)CCC2(CCCN2C(c2nccc3n[nH]cc23)=O)C1 N1(C(c2c(C)sc(O)n2)=O)CCCC2CC12C(=O)O C1(NC(C)=O)CC2(C1)CC1(CC(NC(=O)CCc3cnc(O)[nH]3)C1)C2 c1(C(N2CCC(C(=O)NCC)C2)=O)ccnc(O)c1F C1(C(=O)NC(CCCC)CNC(=O)CCF)CC2CCC(C1)S2 C(=O)(C1=CCCOC1)NC1CCCC(CNC(C(CC)CC)=O)C1 N1(C(c2scc(C(N)=O)n2)=O)CC2CCN(C(c3csc(C(F)F)n3)=O)C2C1 CC(C)CC(C(=O)N(CC(O)CN(C(=O)C=CC1CC1)C)C)C(N)=O c1(NC(CN(C(C(C(C)C)NC2CCCC2)=O)C)C2CC2)ncccc1[N+](=O)[O-] N1(C(C(CCC)C)=O)CCC2(CCCC2C(=O)Nc2cnnc(O)c2Cl)C1 CC(CCCCNC(c1csc(C#N)c1)=O)NC(=O)CC1CCCC(C)O1 C(CS(=O)(=O)CC)OCC.C(C)(CCc1ccco1)(c1nnnn1CCCSC)NCC C(=O)(C1CCCc2nccn21)NCC(C)(C)CNC(C1(CF)CC(F)(F)C1)=O C1(OCC)(CNC(=O)CC2CCCN2C(=O)C(C)(F)F)CN(C)C1 c1(C(N2C(CC)CCC2)=O)cccc(F)c1NC(c1ccc(CN(C)C)nc1)=O c1(NC(CC(C)NC(C(COC)(C)OC)=O)=O)ccc(C)cc1OC c1(OC)cccc(C(C(=O)C2=NOCC2)CC2CCCC(c3ccncc3)C2)c1 C1(O)(CC#C)CCN(C(c2n[nH]cc2CNC(c2sc(CO)nc2C)=O)=O)C1 C(=O)(C1=CC2CCC1C2)N(C1CCC(NC(c2cc(Cl)cnn2)=O)C1)C c1(C(N2CC3N(C(c4ccc(C)cc4Br)=O)C3C2)=O)c[nH]c2cccc(Cl)c12 N1(C(C2N(C)CCN(C(C3CCC(C4CC4)O3)=O)C2)=O)CCC12CCSCC2 c1(C2CCCN(C(C(CC=C)(C)O)=O)C2)ncc2n1CCCC2 c1(SCC(C2CCCN(C(=O)NC(C)C)C2)=O)ccc2c(c1)OC(C)(C)O2 C1(NC(c2c(CC)ccs2)=O)CC2COCC(C1)N2C(C1CC2C=CC1CC2)=O C1(CC)COC(C)(C)CN1C(=O)CCOCCN(C)C(c1cc[nH]n1)=O C(C1CCCN1C)=CC(N1CC(C(C)NC(c2ccnnc2)=O)C1)=O c1(OC)ccccc1C(=O)N(C)CCOCCN(C(=O)C(O)COC1CCC1)C c1(NC(N(CCC)Cc2ccccn2)=O)ccnc(SC(F)F)c1 N1(C(c2cc(C(C)(C)C)no2)=O)CCC(O)C(NC(C2CCOCC2(C)C)=O)C1 C1(CN(C(=O)CC2(C)CCCO2)C)CCN(C(=O)C(F)CC2CCCCC2)CC1 N1(C(COC2C(CC)CCCC2)=O)CCC(CO)(NC(C2C=CCC2)=O)CC1 CC1=CCC(C(N2CC(NC(=O)C(F)(F)C3CCCC3)C(C)C2)=O)CC1 C1(NC(C(CC)OCC)=O)CCC2(CC1)CCN(C(C1CC(C(F)(F)F)C1)=O)C2 c1(CC(N2CC(N(C(CC(C)C)=O)C)C(F)C2)=O)cc(F)cc(Cl)c1 c1(-n2ccc(CNC(=O)NC(c3nc(C(C)C)[nH]n3)C)n2)cccc(Cl)c1 CCCCC(C(=O)NC)NC(C1CC(O)(CNC(=O)Cc2cnc(C)[nH]2)C1)=O CC1CCCC(C(=O)NCC2(O)CN(C(c3snc(O)c3Cl)=O)C2)CC1 C1(O)(CNC(C(CO)OC)=O)CCCN(C(=O)C=CC(=O)NC2CC2)C1 CC1CCc2[nH]nc(C(=O)NC3CCN(C(C4COC(=O)C4)=O)C(C)C3)c2C1 c1(C(N2CCC(CN(C(C(CC)OC)=O)C)CC2)=O)cnn2ccnc(N)c12 c1(SC)ccc(CCC(=O)N(C2CN(C(=O)CC3CC3)CC2F)C)cc1 C(=O)(C(C(=O)NCCCC(C)NC(c1oc(C(C)C)nc1C)=O)C(C)C)OCC N1(C(CC=CC=CCCCCC)=O)CCCC(NCc2ncoc2CC)C1CC c1(C(=O)NCC(C2CCOC2)NC(=O)Cn2cnnn2)cnc2c(c1)CCOC2 c1(CC)cc(=NC2CCCCC2(C)OC)[nH]nc1C(F)(F)F C1(CCCNC(CCN(C)CC)=O)CCCN1C(=O)C(C)(C)c1cnsc1 C1(CNC(COCCCOC)=O)CN(C(c2ncc(F)cn2)=O)CC(C)(C)O1 CC(COC(C1CC1Br)=O)COC(C)(C)C N1(C(CCSc2n(C)nnn2)=O)CC2CCC1CN2C(=O)CNC(=O)C(=O)O N1(C(C(C)C#N)=O)CC2CC(NC(C3CC4(CSC4)C3)=O)C(C2)C1 C1(OC)(CNC(c2csc(C3CCCO3)n2)=O)CCN(C(=O)CCN2CCC2)C1 c1(C(N(C2CCCN(C(=O)CC(=O)NC3CC3)C2)C)=O)cc(F)c(F)c(F)c1F c1(N2C3CN(C(=O)CCCc4ccccc4)CC32)ncnc(O)c1Br C(C(=O)N=c1ccn(CC2CC2)[nH]1)(C1CCC1)NC(C1=NNC(=O)C1)=O CCCC(CCc1ccccc1)C(=O)NCC(C)(C)NC(=O)C1=CC(O)CCC1 N1(C(C(C)N(C(c2ccc(N(C)C)cc2)=O)CC)=O)CCC(F)(CF)C1 c1(C(C)NCCCCCNC)cc(Cl)ccc1OC(F)(F)F c1(C(=O)NCC(CNC(C2(OC)CC2)=O)(C)O)ccn2ccnc2n1 N1(C(c2ccc(CS(C)=O)cc2)=O)CCC2(CCN(c3snc(Cl)c3C#N)C2)C1 C1(CNC(c2nccc(SC)n2)=O)C(C)CCCN1C(=O)CCc1cc(C)no1 c1(N2CCC(C(C)NC(C3CCCCC3O)=O)CC2)cc(Cl)nc(S(C)(=O)=O)n1 c1(CNc2c(C(=O)O)cccc2)cc(Cl)c(F)c(Cl)c1 C(=O)(CCS(N)(=O)=O)N(C)CC1CCCN(C(C2(CC#C)CCCCC2)=O)C1 CON(C)C1CCN(C(c2ccn(CCNC(c3nc(=N)cc[nH]3)=O)c2)=O)CC1 Cc1[nH]c(=NCC(C)NC(C23CC4CC2C3C4(F)F)=O)ccc1C#N C1(C(CNC(C23CSCC2C3)=O)NC(c2cn(C3CC3)cn2)=O)CCCCC1 C(CC(CC)C(=O)N1CCCC1C1CCN(C(C2(C)CC2(C)C)=O)CC1)=CC c1(CCC)ccccc1C(=O)OC(=O)NCC1CCOCC1N(C)C Cc1nn(C)c(N)c1-c1cn(C(C)C(=O)Nc2ccc(CO)c(F)c2)nn1 C(C(O)C(C)(C)CO)N(C)C.C12CCN(CC1)CCNC(=O)O2 Cc1c(C(=O)NCC2CC3CN(C(=O)C=CC(F)(F)F)CC23)sc2nccn12 Cc1cccc(C(=O)NCC2CCC(NC(c3cccc(C4CC4)c3)=O)C2)n1 N1(C(c2c(CCNC(C3(CC)CCCC3)=O)n[nH]c2)=O)CCC2(CC2)C1 CCCCC(CCC)NC(=O)C(CNC(=O)C(C)(C)C1CCCC1)CC1CC1 C1(CNC(CCN(C(c2c(CC)[nH]cc2)=O)C2CC2)=O)CCCC(C)O1 c1(C(N2C(CC)CN(C(C3CN(C(C)C)C3)=O)CC2)=O)ccc(S(C)=O)cc1 C1(C(N(CCCNC(=O)Cc2ccc(O)cn2)C)=O)CCC2CCC(=O)N12 N1(C(C(CC)NC(C)=O)=O)CCC2CN(CC(=O)NCC(F)(F)F)CC2CC1 N1(C(CCC=C=C)=O)CCC2(CCCN(C(c3sc(C4CC4)nc3C)=O)C2)C1 N1(C(C(=O)NCc2c(C(C)C)nc[nH]2)=O)C(C)CCC1C N1(C(COCC(=C)C)=O)CCC(NC(c2cn(CCC)nn2)=O)C(CO)C1 C1(CC)(NC(=O)CS(N)(=O)=O)CCN(C(c2nc(C(F)F)cc(C)n2)=O)CC1 c1(C(N2C(CN(C(c3nc(C)sc3C)=O)C)CCC2)=O)cnc(C2CC2)nc1O CC(C)C(C(=O)N1CCCC1(C)C(=O)Nc1ncc(Cl)s1)c1ccc(F)cc1 n1(CC(=O)N(C2CCCN(CCn3cncn3)C2)C)ccc2ccccc12 N1(C(=O)CCCC(F)(F)Br)CCC2(CC1)CCN(C(c1cnco1)=O)CC2 Cc1cc(F)c(C#N)cc1NC(C1CC(NC(=O)CCn2cncn2)C1)=O C1(NC(CONC(c2c(C)cc(C)s2)=O)=O)CC2CC1CC21CC1 c1(C(=O)NCCC23CN(C(CCCCCC)=O)C(CC2)C3)snc2ccccc12 c1(CC)cc(F)c(C(=O)NC23CCC2CN(C(C2NC(=O)OC2C)=O)C3)cc1F C(=O)(C(=O)N=S(C)(C)=O)NC(C1CCCN1C(=O)Cn1ncc(Br)n1)C C(=O)(CCCCCC#N)NCCC1N(C(Cc2c(C)nc[nH]2)=O)CC(F)(F)C1 c1(C(C)(C)C)nc(=NCC(F)OCCOCCOC)s[nH]1.c1(OCCSC)ccccc1 C12(NC(C=COCC)=O)CCC(CC1)N2C(c1c(Cl)cccc1Br)=O N1(C(c2nc(CCC)oc2)=O)CC2CC(NC(=O)CC3(CSC)CC3)CC2C1 c1(C(=O)NC2C(NC(c3c(C)sc(O)n3)=O)CC2)c(C)ncnc1C C(c1ccccc1C)=CC(=O)NCCC1CCC(NC(c2c(CC)occ2)=O)C1 c1(NC(NC(CC)C)=S)ccc(N2CCC(C)CC2)cc1 Cn1nccc1C=CC(=O)NC1CCCN(C(=O)C(F)(F)CF)C1 C(CC(N)=O)(C(=O)N1CCN(C(=O)CC2CCCCC2)CC1)NC(CC(C)C)=O N1(C(CCc2[nH]c(=N)sc2)=O)CC2CCC(C1)N2C(=O)CNC(c1ccccc1)=O CCCCCC(O)CC(=O)NC1CN(C(c2cc(F)c(C)cc2F)=O)CCC1C C1(C(=O)NC(CCOC)CNC(=O)C2=CCCS2)CSc2ccccc2O1 c1(C(=O)NC2(C)CCN(C(c3c(CC)n(C)nn3)=O)C2)n[nH]c2ccc(C)cc12 c1(SCC(=O)NC2CC(C(C)NC(=O)C(=O)N(C)C)C2)nnnn1C.NC CCCCCCC(F)C(=O)NC(CCNC(c1cnc2n1CCOC2)=O)C(C)C N1(C(c2nc(C)oc2C)=O)CCC(NC(=O)CC(C)C(F)(F)F)C2(CCC2)C1 C1(C(=O)NCC(CNC(c2cc(CO)on2)=O)O)CCN(Cn2cccn2)CC1 CCC(CC(=O)NOCCC(C)O)NC(c1cc2n(n1)CCO2)=O C1(C(N(C2CCOC2)CC#C)=O)CCC2(CN(C(=O)CCc3cncnc3)C2)O1 N1(C(C(COC)N(C)C)=O)CCCCC(NC(C2CC(N(C)C)C2)=O)C1 c1(N(CCS(N)(=O)=O)C)ccnc(NCC2CC2(C)C)n1 c1(N2CC3C(CC)(C3)C2)ccc(S(=O)(=O)NCC2CCC(N(C)C)CC2)cn1 N1(C(C(C2(C)CC2)NC(c2cn(CC)nc2)=O)=O)CCn2ncc(C)c2C1 C(CC(C)C)(C(=O)N(C)CC)NCC=O.c1(C(C(=O)CCC)F)ccccc1 C(C)(C(=O)CN(c1ccccc1)C(C1(O)CCSC1)=O)SC N1(C(C(=O)N(CC(F)Br)C)=O)CCc2nc(C(F)(F)F)ncc2C1 C1(CNC(C(CCC)(C)CC)=O)Cc2ccccc2CN1C(=O)CN(C)C(N)=O c1(CCOC)cc(C(=O)N(CC(C)NC(C2CC(C#N)C2)=O)C)no1 C1(N(C)C(C2(c3cncnc3)CN(C(=O)OC(C)(C)C)C2)=O)CCCSC1 c1(CN(C)Cc2cc(OC)c(Br)c(OC)c2)ccc(N)c(C)c1C N(S(=O)(=O)N1CCCC1)C(c1ccc(Cl)cc1)C(C)C.C1(=O)CO1.C1CO1 c1(C(=O)OC)ccc(C)nc1NC(C1(C)CCCN(C(c2cc(C)[nH]c2C)=O)C1)=O N1(CCNC(C(CC)CC)=O)CCCN(C(C2(c3n[nH]cc3C)CC2)=O)CC1 C1(CC(N2CC(NC(=O)C=Cc3cnc[nH]3)C(F)CC2)=O)CCC2(CC1)COC2 C1(F)(C(C)C)CCN(C(=O)C(C)(C)NC(=O)CCCOc2ccccc2Cl)C1 C1(C(C)(C)C)CN(CC23CCCC2CC(=O)N3)c2ccccc2O1 N1(C(C=Cc2c(C)noc2C)=O)CC2CC1CN(C(=O)C(C)C(F)(F)C(F)F)C2 c1(C(=O)Oc2cc(OC3CCCC3)cc(F)c2)cccc(O)c1[N+](=O)[O-] c1(CC(=O)NCCNC(C2(COC)COC2)=O)ccc(SC)cc1 c1(C(N2CCC(N(C(c3cc(C)oc3)=O)C)C(C)C2)=O)cc(N)c(Cl)c(O)c1 Nc1c(C(N2CCN(C(c3cccc4nncn34)=O)C3CC23)=O)cc(F)cc1Cl Cc1csnc1C(=O)N(CC(Cc1ccccc1)NC(c1cncs1)=O)C C(C)(C)(CC(F)C(=O)N1CCC(C(F)F)CC1)NC(C(C)CN(C)C)=O c1(N(C2(c3n(CC)nnn3)CCCC2N(C)C)C2CC2)cc(C2CC2)ccc1F c1(COC)nc(NC2CCS(=O)CC2)cc(=NC(C)c2nncs2)[nH]1 c1(CNC(C2CCC(n3cc(CC(CO)CO)nn3)CC2)=O)ccnc(O)c1Br c1(C(=O)NC(CC)CNC(=O)CC2CCS(=O)(=O)C2)c(C)cccc1N CC(C)C(C(=O)NC(C)C(=O)NO)NC(=O)CN1CCNC(=O)C1 N1(C(C23CCC(OC)(CC2)C3)=O)CCC2CN(C(=O)CC(C)C(C)(C)C)CC12 c1(CNC(N(C)Cc2c(OC)n[nH]c2)=O)cc2c(Br)c(F)ccc2[nH]1 C(=O)(C1CCc2cccnc21)NCC1(O)CN(C(C2CCCC(=O)CC2)=O)C1 C(=O)(C(O)CCCCC)NCC(N(C(CCC(=C)Br)=O)C)C1CC1 C(CCCC(=O)NC1(CCCNC(=O)C(C)(C)N2CCCCC2)CC1)OC C1(NC(c2c(C=C)cccc2)=O)CCC2(C1)CN(C(=O)C(C)OC)C2 C(=O)(C1=CCCSC1)N1CCC(N(C(c2oc(C)nc2C)=O)CC)C1 N1(C(CSCCN(CC)CC)=O)CCC2(CC1)CC2NC(=O)CNS(N)(=O)=O N1(C(CC(C)SC)=O)CCCC(N(C(=O)CCCC2CCC2)C)C1 c1(SC(c2ccc(F)cn2)C)nc2ncccc2s1 c1(N2C(C(=O)Nc3cnc(OCC)nc3C)CNCC2)ncnc2c1cnn2C N1(C(CCNC(C)=O)=O)CC(C2CCCCN(C(C3CCC(C)CC3)=O)C2)C1 c1(CC)nn[nH]c1C(=O)NCCn1ccc(C(=O)NC2CC2F)c1 C1(C(C)C)CCN(CC(=O)NCc2cccc(Cl)c2)CC1 C1(C(=O)NCC(CC=C)NC(=O)CC2(COC)CC2)CCCN1S(=N)(=O)N(C)C c1(N)ccc(ON)nc1.c1(C(CNC2CCOCC2)OC)ccc(Cl)cc1 c1(C(=O)NCC2C(C)CCN2C(=O)CC2CC2)cccc2c1COCCN2 N1(C(=O)OC(C)(C)C)CC2C(C(=O)NC3CCC3CNC(c3cnsc3)=O)C2C1 C(=O)(CC(C)(C)CC(F)F)N1CC(NC(CSc2n(C)nnn2)=O)C2C(C1)C2 C(=O)(CCC1=NNC(=O)CC1)NCC1(F)CN(C(c2ccc(C)c(Cl)c2Cl)=O)C1 C1(C(=O)NC2CCCC(CNC(c3cnn(C)c3Cl)=O)C2)COC2(CCC2)CO1 C1(NC(c2ccncc2F)=O)CN(C(=O)Cc2cncs2)C2CCCC12 c1(C(=O)NC(C2CCN(C(c3coc(C(F)(F)F)c3)=O)C2)C)cccnn1 N1(C(C2(O)CCC(C)CC2)=O)CCC(F)(F)C(CNC(c2cnccc2Cl)=O)C1 c1(C(=O)NC(C(C)(C)O)C(=O)O)ccc2c(c1)nc(O)n2C1CC1 N1(C(COC(C)C)=O)CCC2(NC(c3cc(C(N)=O)cs3)=O)CCCCC12 C1(CC(=O)NCC(CNC(C=CC)=O)(C)OC)CCOCC1(C)C C1(NC(C2N(CC)CC2)=O)CCN(C(=O)C(C)(C)CC2CCOCC2)CC1 c1(OC)cccc(CCC(N2CC(C(=O)NC(C)C)CC(F)C2)=O)c1C CC1(C)CC2(CC2C(N2CCOCC2CCNC(=O)COCC2CCOC2)=O)C1 Cc1ccc(C(=O)NC2CN(C(c3ccc(F)c(F)c3)=O)CC2C)c(O)n1 Cc1cc2cc(C(=O)NCC3CCCN(C(C4CCC4C)=O)CC3)oc2cc1C C(=O)(C(C)CNC(=O)CC(Cl)Cl)N(C(c1cccs1)C)C c1(CC(=O)NCC(c2ccccc2)NC(CCOCC#C)=O)ccn(C(F)F)n1 C1(NC(CC(CC)OC)=O)CC2CN(C(c3cc(C(C)C)nc(O)c3)=O)CC12 c1(C(=O)NC(CCF)C(=O)NCc2cc[nH]n2)ccc(F)cc1F C1(NC(=O)COC2CCCCC2)CCN(c2nnnn2C2CCC2)CC1O Cc1cc(C#N)ccc1C(N1CCC2CCCC12C(=O)NCC(C)O)=O n1(CCC(=O)NC2CC(C)(NC(CC(CCC)O)=O)C2)cc([N+](=O)[O-])nc1C C=C(C)CCCC(=O)N(C1CCN(C(c2ccsc2CC)=O)C1)CCC c1(CC)ccc(C(=O)NC2CC2NC(C2CCCCN2C(C)C)=O)c(F)c1 c1(C(=O)NCC(C2CC2)Nc2cc(OC)ncn2)n[nH]c2cc(C)ccc12 C1(NC(CCCC#CC)=O)COC2(C1)CN(C(c1ccc(C#N)cc1)=O)C2 N1(C(C2C(C)C2C)=O)CCN(CC(=O)NC2(CC#C)CCOC2)CC1 N1(C(C(n2c(C)ncc2)C)=O)CCC(O)(CCNC(=O)C(C)N(C)C2CC2)CC1 C(=O)(C(C)(F)CCCC)N1CC(O)(C(C)NC(C(C)=C2CCC2)=O)C1 C1(NC(CCSCC)=O)CCCC(NC(=O)C=CCc2ccncc2)C1 c1(C(=O)NCC2CCN(C(c3[nH]cc(C)c3)=O)CC2)csc2nccn12 N1(C(C2(CCCC)CC2)=O)CC2CS(=O)(=O)CC2(NC(c2ccnnc2)=O)C1 C(=O)(CC1=NNC(=O)C1)N(C)CCNC(C1(C)CC1F)=O c1(OC)ccc2c(c1)C=C(C(=O)N1CCC(CN(C(C3CC3F)=O)CC)C1)CO2 C=CC(CCC)CC(=O)N1CCC(C)C1C(N1CCOC(C)(C)C1)=O CCCCCCC(=O)N1CCOCCC1C(=O)N(C)Cc1nc(CC)no1 c1(C(=O)NC(CC)CNC)ccc(CSC)o1.C1(=O)CC12CC2.N(C)(C)C N#Cc1cncc(NC(C2CN(C(C3CCC(=O)N3)=O)CCC2O)=O)n1 N1(C(c2ccc(SC)s2)=O)CC(NC(C2CCCC(CF)C2)=O)C2(CC2)C1 C1(NC(C2CN(C)C2)=O)CC(C(=O)NC23CC(C)(C2)C3)C12CCC2 C(C)(C)(CC(C)NC(c1cc(CNC(c2cc(C(N)=O)[nH]n2)=O)[nH]n1)=O)OC N1(C(CSC)=O)CC(NC(c2nnn(-c3cc(C)ccc3C)c2C)=O)C(C)(C)C1 C(CCC(=O)N(CCSC)CC)(C(C)C)NC(CC(CC)OC)=O C12(C(=O)NCCCCC(=O)NCC(C3CCC3)OC)CCCC(CO1)C2 C(=O)(C1CCCc2nccn21)NC12CC(NC(CN(S(N(C)C)(=O)=O)C)=O)(C1)C2 c1(C(N(C)CC2CCN(C(CCCC(C)C)=O)C2)=O)ccc(Cl)c(Cl)c1N N1(C(C(C=C)O)=O)CCCC1(C)CCC(=O)NCc1ccoc1C Cn1cnc(N)c1C(N1CC(c2ccc(F)cc2)C(N)C1)=O c1(C(N2C(CNC(C=CC)=O)(COC)CCC2)=O)cn2ccc(Br)cc2n1 Cc1ncc(Cl)c(C(=O)NC2CC(NC(=O)CN3CCSCC3)C(O)C2)n1 C1(O)(CN(C)C(N)=O)CCN(C(=O)C(C(C)O)NC(c2cc(C(N)=O)co2)=O)C1 C(CN=c1[nH]c(C(=O)N(C)C)cs1)c1scc(C)n1 c1(C(C2CC2)NCC(C)OC(F)F)cc2cc(Br)cc(F)c2o1 C1(C(C(=O)O)F)CCN(C(=O)COC2CCOCC2)C1 N1(C(C(C)OCCCC)=O)CCC(NC(c2c(OC)cccc2CC)=O)C(C)C1 C1(C(=O)NCCC(Cn2cc(C(C)OC)nn2)F)CCc2c(cnn2C)C1 C1(CNC(C2CN(C)C(=O)N2)=O)CC2(CO1)CN(C(c1ccoc1)=O)C2 N1(C(CCCn2cc(C(CSCCOC)C)nn2)=O)CC(C)=C(C)C1 n1(CCCOC)cc(C(=O)O)nn1.c12csc(n1)CNC2=O CCC(CC)C(F)C(=O)NC1(CNC(c2ccc(OC)nn2)=O)CCOC1 C1(C2(NC(CC(=C)C)=O)CC2)CCCCN1C(c1cnn(C)c1COC)=O C1(CCNC(CCN(C)C(=O)C2CC2)=O)CCCCN1C(c1[nH]ncc1C#N)=O Cc1cc(C(N2CCC3CC23C(=O)NCCN(C)C)=O)cc(O)n1 c1(C(=O)NC(C)(CNC(c2nnn3c2CCC3)=O)CO)ccc2cnoc2c1 c1(C(N2C(C)(C(N3CC(C(=O)OC)OCC3)=O)CC2)=O)ccc(Br)c(C)c1F c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C(C)C2)ccnc(O)c1Br C1(CNC(c2cc(SC)no2)=O)C2CN(C(=O)C(c3ccccc3)N(C)C)CC12 Cc1ccccc1S(=O)(=O)CC(=O)N1CCN(C(C2CCC(O)C2)=O)CC1C N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2(CC(C(=O)N3CCCC3C(N)=O)=NO2)C1 C1(C(=O)NCC(NOCCCOCC)=O)COCC(C)O1 n1(CC)c(C(=O)NC(C)(CO)C(=O)NC2CCCOC2)cnc1O N1(C(C(CCCOC)C)=O)CCc2ccc(C(=O)N(CC(C)(C)C#N)C)nc2C1 C(=O)(CC(C)(O)COC)NC1(C(N2CCCC(OC)C2)=O)CSC1 N1(C(CC(C)OC)=O)CCCC(NC(C2(F)CC2)=O)C1 Nc1cc(C(=O)NC2CN(C(=O)C(c3cccc(Br)c3)(F)F)C2)cc(F)c1 c1(C(N(CCOC)CCNC(c2c[nH]nc2SC)=O)=O)cc2cccc(F)c2o1 CC1(NC(C2COCC2(C)C)=O)CCN(C(=O)COC2CC(F)(F)C2)CC1 N1(C(C2CC(C)(NC(C(CSC)O)=O)C2)=O)CCC(F)(CO)CC1 c1(C(C(=O)NC2C(NC(Cc3cc(COC)on3)=O)COC2)O)cccc(F)c1 c1(C(N2CCC(NC(COCCC)=O)C2)=O)cc(S(C)(=O)=O)c(Cl)cc1Cl CC1CN(C(c2ccnc(C#N)c2)=O)CCCN1C(=O)C(N1CCN(C)CC1)C c1(C(=O)NCCC(CNC(c2nn(CC)c(C)c2)=O)O)ccc(=O)n2c1CCC2 Cc1cc(CNCc2cnc(-c3cccs3)s2)c2[nH]c(C)c(C)c2c1 c1(C(N2CCC(CC(=O)NCCCF)C2)=O)cccn2ccnc12 c1(C(=O)O)ccc(Cl)c(S(=O)(=O)Nc2ccc(O)cc2)c1 CC1CC(NC(=O)C(F)=CCCF)CN(C(c2cnn(CC3CC3)c2)=O)C1 C(=O)(CS(=O)(=O)Cc1cccs1)NC1CCC(NC(C2(C)CCCS2)=O)CC1 c1(C(=O)NCC(C(C)C)NC(c2cc3cccn3cn2)=O)ccc2nncn2c1 c1(C(N(CC(C)NC(C(CC)OC2CCCC2)=O)C)=O)cc(N)cc(O)n1 Cc1cc(C)cc(C=CC(=O)NC2CC(NC(C3CCC3F)=O)C2)c1 c1(CC)nn(C2CC2)cc1C(N1CCOCC1CNC(C12CCC(C1)C2)=O)=O Cc1cc(CN(C(=O)NC2(C)CC2C(=O)O)C)cc(C)c1Br C12(C(=O)O)CCCOC1CN(C(c1ccn3cccnc13)=O)C2 c1(OC)ccc(NC(=O)C(c2ccc(Cl)nc2)N(C(CO)C(C)C)CC)c(C)c1 c1(C(=O)NCC(C)(CC(C)C)NC(c2c(C)cc[nH]2)=O)ccc2c(c1)OCO2 C(=O)(C(C)CS(C)=O)NCC(C)CN(C)C(c1ccnn1C1CC1)=O C1(n2cc(C(C)OC)nn2)CC2CCC1(NC(=O)CCOc1ccccc1)C2 Cc1cc(C(=O)NC(C2(O)CN(C(=O)C(C)Sc3ccccc3)C2)C)ccn1 C(=O)(C(C)(C)C(C)C)NC(C(C)C)CNC(=O)Cc1scnc1-c1cccs1 N1(C(C2C(C)=C2)=O)CC(NC(c2nn(C)c3c2CCCC3)=O)CC12CCOCC2 C1(C)(CNC(C2CC(CCC)C2)=O)COCCN(C(c2cnn(CCC)c2)=O)C1 c1(COC)ccc(C(N2CCCC2(C)C)C(=O)NC2CCCC2)cc1 C(=O)(C(O)C(C)(C)C)N(CCNC(C=Cc1cn(C)nc1)=O)C1CC1 c1(C(=O)NCC=CCNC(CCSCC(N)=O)=O)cnoc1-c1ccc(Cl)s1 C(=O)(C(C)(C)CCCO)NC1CN(C(c2cc(CC)[nH]n2)=O)C(C)CC1 Cc1cc(F)ncc1C(=O)NCCC(C)N(C)C(c1cc(C(F)(F)F)cs1)=O c1(NC(C(C(=O)OCC)CC)=O)cccc2c1CCN(C(=O)CSC1CC1)C2 S(=O)(=O)(c1c[nH]ccc1=NC1CCCC(CO)C1)N(CCC1CC1)CC N1(C(CCCOCCC)=O)CCN(C(c2cccc(O)n2)=O)C(CC(F)(F)F)C1 C(CN(C)C)(N=c1ccnc(NC(c2csnn2)C)[nH]1)c1c(OC)cccc1 CC(C)CCCC(C)C(=O)NC1CC(C(N2CCOCC23CC3)=O)C1 CCCC(C#N)C(=O)N(C)CC1CCCN1C(c1ccc(C(C)(F)F)nc1C)=O Cc1cc2ccc(C(=O)NCC(C)(O)CNC(c3nc(C4CC4)cs3)=O)cn2c1 CN1CC(O)CCC1C(=O)NCCCC(=O)N1CC(N(C)CCO)C1 c1(OC)cc(OC)nc(C(=O)NC2(C)CN(CC3CCC(=O)NC3)C2)n1 C1(NC(C(CC(=C)Cl)NC(=O)C(C)CC=CCC)=O)CCn2cncc2C1 Cc1ncc(NC(C2CCCCN2C(=O)C(C)NC(c2ccc[nH]2)=O)=O)cc1Br CCC(CCCO)NC(=O)CCN(C)C(C1(CO)CCCC1)=O c1(C(=O)NC(CNC(C(C)Cn2cccn2)=O)CO)cc(Cl)cnc1O C1(NC(C(=O)NC(C)CN2CCOCC2)=O)CCCC2CNCC12 N1(C(Cc2c(Cl)cn(C)n2)=O)CCCCC(CNC(=O)CCCc2cnn[nH]2)C1 CC#CCC(C(=O)Nc1ccccc1O)NC(C1CC1(F)F)=O C(=O)(C(C)S(C)(=O)=O)N1C(CC)C(C(=O)NC(c2ncnn2CC)C)CC1 C1(C)(NC(N2CCC(C(=O)Nc3ccn(C4CC4)n3)C2)=O)CCN(C(C)(C)C)C1 c1(C(=O)NC2C(CNC(C(CCSC)OC)=O)CC2)ccc2nnn(O)c2c1 c1(OC)ccc(CCC(N2CC(C)N(CC#N)CC2C)=O)cc1[N+](=O)[O-] C1(CC(N2CCCC(NC(c3on(C)c(=O)c3)=O)C2)=O)CCC2(CC1)OCCO2 C1(CNC(C2CC(OC)C(OC)C2)=O)CC2(CCN(C(=O)CSC)C2)CO1 C1(CN(CCCNC(C(C2CC(F)(F)C2)OC)=O)C2CC2)CCCC(F)(F)C1 CC(CC(=O)N(C1CCC(NC(=O)CCC(F)(F)F)CC1)C)CC(C)(C)C C1(NC(=O)CC2CC=CC2)CN(C(=O)CCSCc2ccccc2)C2CC12 C12(C(=O)NCCn3cc(C(=O)NCC(C(C)C)(C)F)nn3)CCC(CC1F)C2 C(CCCCC(=O)NCc1cccc(CO)n1)N(C(C1C(C)CCCC1)=O)C C(=O)(C1OCCc2ccc(C)cc21)N(CCNC(=O)C(C)(C)O)CC N1(C(C(C)=O)=O)CCC(C2CCCN2C(=O)CSc2nncs2)C1 c1(OC)cccc(C(=O)NC23CC2CN(C(c2cncc(Br)c2)=O)C3)c1F N1(C(C(C2CC2)OCC)=O)CC(CO)C2(C1)CN(C(=O)COC1CCCC1)C2 c1(CN(CC(C(=O)O)OC)C(C)C)ccc(Cl)cc1C CC(C)C(C)C(=O)NCCCC1(NC(=O)C(c2ccc(F)cc2)C)CC1 N1(C(C2C3CN(C(CN(C(COC)=O)C)=O)CC32)=O)CC(C(C)C)CCC1C c1(CNC(=O)NC(c2ccccc2)C)ccc(-c2ccccc2)cc1F c1(C(=O)NCC(C2CC2)N)cccc(CO)n1.N1(C(C(=O)NC)=O)CC(O)C1.CF C(=O)(CCCCN=[N+]=[N-])NC1(CNC(C2CCC(CC)O2)=O)CC(OC)C1 C1(C)(NC(C(C)OC(c2cccc(N3CCCC3=O)c2)=O)=O)CCNC(=O)C1 S(=O)(=O)(c1cccnc1N(C)Cc1nncs1)N(C(C)C)CCO c1(C(N2CCC(CN(C(C(CC)NC(C)=O)=O)C)C2)=O)cccc(Cl)c1 c1(NC(CN(C(=O)CC(C)N(C)C)CCC)=O)cccc(-c2nn[nH]n2)c1 O=C1Cc2cnc(N3CCCC34CN(Cc3ccc([N+](=O)[O-])o3)C4)nc2N1 C1(C2CN(C(=O)CNC(c3ccccc3Cl)=O)C2)(NC(CC(CC)OC)=O)CC1 C(=O)(C(F)C(C)C)N1CCC(C(C)(C)NC(C=CSC)=O)C1 Cc1ccccc1NC(C1CN(C(C2C(C)(C)C2(F)F)=O)CCO1)=O C1(C(=O)NOc2nc[nH]n2)(NC(c2cn(CC)nn2)=O)CCN(C)C1 C1(N(CCNC(c2ccc(Cn3ccnc3)o2)=O)CC2C=CCC2)CCOCC1 c1(CC)nc(=N)[nH]c(=NCC2(CNC(C34CCCCC3OCC4)=O)CC2)[nH]1 CC1CN(C(C2CCN(C)CC2)=O)CCC1CNC(C1Cc2nccn2C1)=O N1(C(c2nc(Cl)cs2)=O)CCC2(CCCN(C(C3(N(C)C)CCSC3)=O)C2)C1 c1(C(N2C(C)CCC(CNC(=O)CN=S(C)(C)=O)C2)=O)cc[nH]c2nccc1-2 C1(C(=O)NC2CC(C)(CC)OCC2)CC2C=CC1N(C(C1CCCN1CC)=O)C2 n1(CC)nccc1NC(=O)C(c1nc(C(=O)Nc2cn(C(C)(C)C)nn2)cs1)C C(C1=Cc2ccccc2OC1)=CC(=O)NC1CCN(C(C2CCCSC2)=O)CC1 c1(C(N(C2CCN(C(=O)C(c3cncn3C)O)C2)CC)=O)ccc(CN(C)C)[nH]1 c1(OC)cncc(CNC(C2CC(CO)N(C(c3cccc(O)c3)=O)C2)=O)c1 CC1CC(C(=O)NC2CCCN2C(=O)C2CC2)N(C(=O)CN2CCC(C)C2)C1 CC(CO)(CO)C(=O)N1CCC(NC(c2cccc(C(F)F)c2)=O)C1 CC1CCCC(CC(=O)NC2(C)CN(C(c3snc(O)c3Cl)=O)C2)O1 c1(OC)ccnc(CNC(=O)CN(C(C2CC(C(C)C)C2)=O)C(C)C)c1 c1(C(=O)NCCC2CCN(C(C(CCC)C)=O)C2)cc(C(F)(F)F)cc(Cl)c1 C1(NC(C2(CCN(C)C)CC2)=O)CC2CN(C(C3CC4COCC4C3)=O)CC2C1 N1(C(COCCSC)=O)CCC2CCCC12CNC(=O)CN1CC(C)(C)C1 C1(NC(c2c(CC)noc2)=O)CC12CCN(C(=O)CCOCCOCCO)CC2 c1(OC)cc(S(=O)(=O)N2CCCC2)ccc1COC(=O)CCCCC1CC1 c1(C(=O)NCC(C2CCC2)NC(C2C(C)(C)C2(F)F)=O)coc2c1C(=O)NCC2 n1(CC(=O)NC(CNC(c2c(CC)n[nH]c2)=O)C(C)(C)C)c([N+](=O)[O-])cnc1C C#Cc1cc(C(N2CCC(NC(C3(CC4CC4)CC3)=O)C(C)C2)=O)cc(N)c1 c1(C(=O)NC(CNC(c2c(C)nn(C)c2)=O)C(C)C)ccc2c(Br)cnn2c1 CC1C(=O)CCC(NC(=O)Nc2cccc(N3CCCC3)c2)C1 N1(C(CC(C)C)=O)CC2CC(NC(c3c(F)ccc4occc34)=O)CC1C2 N1(C(C=C(COC)C)=O)CCCCC1CCN(C)C(C1(c2ccncc2)CC1)=O C1(C(=O)NC2(C)CN(C(=O)CCc3ccc(N)cc3)C2)Cc2ccccc2CO1 C(CCCCC(=O)N(CCC(C)NC(=O)C(C1CC1)N(C)C)C)SC Cc1ccc(C(=O)NC(Cn2cncn2)C(=O)NCc2ccnc(CO)c2)cn1 c1(C(=O)NC(CN(CC(C)NC(c2ccon2)=O)C)C)ccccc1 CC1CC(F)(F)CCN1C(=O)CC1CC2CCC(C1)N2C(C1CC1(F)Cl)=O N1(C(c2cc(C)cc(C)c2)=O)CC2(CCC(CNC(=O)CCNC(=O)CO)O2)C1 O=[N+]([O-])c1ccc2c(c1)OCC2NCC(C1CCOC1)N1CCCC1 C1(N(C)C(C2CC2C(C)(F)F)=O)CCN(C(c2cnc(S)nc2)=O)CC1 N1(C(c2nc(CC)oc2C)=O)CCN(C(=O)CC23COC(CC)(C2)C3)CC12CC2 N1(C(CCC(=O)OCC)=O)CCC2(CC(NC(=O)CCC3(C)CC3)CO2)C1 Cc1cc(C2(O)CN(C(C3C(C(=O)OCc4ccccc4Br)C3)=O)C2)cc(C)c1 Cc1noc(C)c1C(=O)NCC12CC1CN(C(=O)COc1ccccc1F)C2 C1(C(=O)NCc2cn(-c3cc([N+](=O)[O-])ccc3Br)nn2)CSC(c2cccs2)=N1 C1(C(=O)NC(CC=C)CO)(C(C)C)CCN(C(=O)COCc2nc(C)no2)CC1 N1(C(CC(c2ccccc2-c2nn[nH]n2)C)=O)CCC(C2CCNCC2)CC1 Cc1cnc(COCCC(=O)NC2CC2NC(C2CCCO2)=O)[nH]1 Cc1cccc(NC(=O)NC2CN(C(=O)C(c3c(F)cccc3F)(F)F)C2)c1F N1(C(C2C(C)(C)C2NC(=O)CC2CSC2)=O)CCN2CC(F)CC2C1 C1(C(=O)NC2(CNC(c3cncc(C4CC4)c3)=O)CC2)CCCS1(=O)=O CC1(C)CCN(C(=O)C(C2CCCCC2)=O)C(C(N2C3CCCC2COC3)=O)C1 c1(C(C)(F)F)cc(C(=O)NC2CC(NC(C3CC(F)(CF)C3)=O)C2)[nH]n1 CC1CN(C(C2CC(=O)NC2(C)C)=O)CCC1NC(=O)Cc1coc(C(F)F)n1 CCCN=C1NOC2CC(N1)C21CCC1.c12ncccc1NC2=O.C(C)(C)OC c1(C(=O)NCc2cn(-c3ccc(OC)c(F)c3)nn2)cccc2c(Br)cccc12 c1(C(=O)NC(C2CCCCC2)c2nn[nH]n2)cc2c(Cl)c(Cl)ccc2[nH]1 C1(C(=O)NCC2(C)CCCNC2)CC(C2CCC2)C1 CCC(C)(C)C(O)C(=O)N1CC2CC2(C(N2CCN(C3(C)CC3)CC2)=O)C1 Cc1cc([N+](=O)[O-])ncc1C(=O)NCCCCNC(C1(C)C=CCC1)=O C12(C(N3CCCC(NCCCC)C3)=O)COCC1CN(C(=O)C(O)COC)C2 c1(NC(c2c(C)nc(C)c(C)n2)=O)cnn2c1N(C)CCC2 c1(C(N(C2CCCCN(C(c3coc(Cl)n3)=O)C2)C)=O)ccn2cccc2c1 C1(C(=O)NC(CCSC)C(=O)NC(c2csc(C)n2)C)Cc2ccccc2C1 C(C(CC(=O)NC1(CF)CCN(C(c2ccoc2)=O)C1)C(F)F)N(C)C C(=O)(CC(C)CCCCCCCCCCC)NCC=C.C(C)(C(C)(C)N)NC(CC=C)=O N1(C(c2cc(CC)n(C)n2)=O)CCC2(CC1)CCN(C(=O)C1=NOCC1)CC2C N1(C(C(C)OCCN(C)C)=O)CC(NC(c2ccc(OC(C)C)nc2)=O)C(C)(C)C1 c1(C(=O)NC2(CNC(C3CC=C(C)CC3)=O)CCOC2)cccc2nn(C)cc12 c1(C(=O)NCC2(F)CC(CNC(c3c(C)cccc3)=O)C2)c(N)cc(Cl)nc1Cl c1(OCCC(=O)NC(C(C)(C)NC(C(CCC)C)=O)C)cccc([N+](=O)[O-])c1 C1(NC(CC(C)n2ccnc2)=O)(CO)CCCN(C(=O)C=CC(=O)N(C)C)C1 c1(NCc2c(C)scc2)cc(=NC2CCC(C)C2)[nH]c(C(C)C)n1 c1(C(N2C(CC)CC(C)CC2)=O)nc2sc(C)cn2c1C Cc1cc(C(N2CCC2CNC(=O)Cc2ccc(Cl)cc2)=O)nn1C Cc1ccc(-c2cnc(C(=O)N(CCC(C)C)CCO)c(C(F)(F)F)c2)c(C)n1 Cc1ncc(C(=O)NC(C2(CNC(C3CN(C)CCO3)=O)CC2)C)cc1N C(=O)(CS(=O)(=O)CCO)NC(C1CCOC1)CNC(c1cc(C)nn1C)=O C1(CC)CN(C(=O)CC2CC(OC)C2)CCN1C(=O)Cn1nc(O)ccc1=O c1(C2C(C(N3C(C(C)NC(CC)=O)CCC3)=O)C2)cncc(F)c1 N1(CC(c2ncn(C)c2)O)CCN(C(c2cc(C3CC3)ncn2)=O)CC1 c1(C(N2CC3C(NC(c4n(C)c(Cl)cn4)=O)C3C2)=O)cc(Cl)c2ccccc2n1 S(=O)(=O)(c1ccc(C(C)=O)cc1)Nc1c(OC)ccc(C(C)(C)OC)c1 Cc1coc(C)c1C(=O)NCC1CCC(N(C(=O)C(C)CC2CCCC2)C)CC1 c1(OC(C)C)cccc(C(=O)OC(C)(C)C)c1.C(=O)(CCOC)N1CCOCC1 C(CCC)(C(O)C(=O)NC(C)(CC)C(C)(F)F)NC(CCCCCC)=O N1(Cc2cc(C)ncn2)CCC(NC(=O)Cc2ccc(C3CC3)c(C)c2)C(C)C1 CC(C)C(C(=O)N1CCC(Cc2cn(C3CCCCC3)nn2)CC1)C(C)C N1(C(CC(C)F)=O)CC(F)CC1CN(C(=O)CCCc1cccc(Br)c1)C C1(NC(CC(=O)OC)=O)CCCN(C(c2cc(C)[nH]n2)=O)C1CO c1(C(N2CCN(CCN(C(C(=O)NCC)=O)C)CC2)=O)cccc2occc12 c1(C(N2CC(C(=O)NC)OCC2)C(=O)NCCCC2CC2)ccc(OC)cc1F c1(OCC(=O)NCC2(NC(=O)Nc3nc[nH]n3)CCC2)ccc2c(c1)CCC2 Cc1nc(C(N2CCC(CC(N3CCC(C4CC4)C3)=O)CC2)=O)ccc1C#N C=CC1CCCN(C(=O)C(CC(C)C)NC(c2cc[nH]c2CCC)=O)C1 CC1(C)CC(C(N2CCOCC(NC(c3cnoc3)=O)C2)=O)CCO1 C1(NC(COCC)=O)CC2CN(C(=O)COc3ccc(C)cc3C)CCN2C1=O S(=O)(=O)(c1ccc(Cl)cc1)N(C1CCCC(C)C1)CCN1CCc2sccc2C1 N1(C(CN(C(CCCCC)=O)CC)=O)CCC(NC(=O)C(F)=CC2CC2)C(F)C1 N1(C(C)C)CCC(NC(=NCCN)NS(=O)(=O)c2cnn(C)c2)C2OCCC12 Cc1ccc(C=CC(=O)OCC(C2CCC23CCC3)=O)o1 C1(CCC)CN(C(=O)COCCF)CCN1C(=O)C(C)Cc1cccnc1 C(=O)(C1=C(Cl)CCC(C)C1)N1CC(NC(CC2(OC)CCC2)=O)C(OC)C1 N1(CCC(=O)NCCN(C(=O)C=CSC)CCC)CCSC(C)(C)C1 Cc1nccc(C(N2CCC(F)(CNC(c3ccc(Cl)s3)=O)C2)=O)n1 C(=O)(CCC(C)CN(C)C)NC(C1CCN(C(=O)C(C)(C)CO)CC1)C C(CC1CCC1)(C(=O)NCCC1CC(O)C1)NC(C1C(=C)C1)=O C(CCC(C)(C)NC(C1CCCC1O)=O)NC(C(c1ccccc1Cl)N(C)C)=O C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CC(CNC(CCC#CC)=O)C(O)C1 Cn1nc(Cl)cc1NC(c1sccc1CNC(C1CCC(=O)N1)=O)=O c1(C(N2CC3C(C(=O)NC(CC(C)C)CO)C3C2)=O)cnc2cc[nH]c2c1 c1(C(=O)NCCC2N(C(c3c(C)nccc3)=O)CCSC2)ccc(Br)c(F)c1C C(CC(=O)NCC1CC(=C2CCC2)C1)(C(F)(F)F)NC(C=C(CC)CC)=O C(=O)(C1=Cc2ccccc2C1O)NCCC1(O)CN(C(C(CC)(C)F)=O)C1 C(=O)(C(C)(CNC(=O)CC(=O)NCC#C)CC)NC(CC=C)C1CC1 n1(C(C)C)ncc(Cl)c1C(=O)N(C(C)CNC(=O)CCCCc1cnc[nH]1)C c1(C(=O)NCC(CN(C(c2cnc(C(=O)OC)s2)=O)CC)(C)C)cccc(SC)c1 c1(OCC)cc(CN2CCN(C(=O)CCC=CC(C)C)C(CC)C2)ccc1OC C(c1ccco1)=CC(=O)NCC(COC)NC(=O)C(C)OC1CCOC1 CC1CCC(C)(C(=O)NC2(CN(C(=O)CCSCCC#N)C)CC2)CC1 N1(C(C2(C#N)CCCC2)=O)CC2CC(NC(C3CCC3(F)F)=O)C1C2 C1(CNC(C(CC)(C)CO)=O)CN(C(c2scnc2C(F)F)=O)CCC1(C)C c1(C(N2CCC(CNC(C(C)CSC(F)(F)F)=O)C2)=O)cc(N)cc([N+](=O)[O-])c1 C(=O)(CCC(C(C)C)NC(=O)Cc1c(C)n[nH]c1C)NCCC(=O)NC(CC)C c1(C(=O)NC2CCCN(C(C3C(C)C3)=O)C2C)cncc2c1CCNC2=O c1(CC(=O)NCCCN(C(C2CN(CC)C(=O)C2)=O)C)cccc2c1OCCC2 N1(C(c2c(CC)csc2)=O)CCCN(C(C2CCOC(C)(C)C2)=O)C(CO)C1 c1(NC(=O)NC2(CC#C)CCCOC2)cc2ccncc2[nH]1 c1(C(=O)NCC2OCCCN(C(C3OCCN(C)C3)=O)C2)cnc2[nH]ccnc1-2 C(C1C(=O)N1)OC.c1(C(N2CCC(OCC3CC3)C2)=O)cn(CC(N)=O)nn1 c1(C(=O)NC2CN(C(c3nn[nH]c3Cl)=O)C2)cnc(C2CC2)o1 N1(C(c2[nH]cc(C)c2)=O)CC(C(=O)NCC2(C)CC3CCC2C3)CC1(C)C CC(C)(CC(=O)N1CCC2C(NC(=O)C=CC3CCCC3)C2CC1)CC(F)F C12(CC)CN(C(=O)COCCF)C(CNC(=O)CN3CCSCC3)(C1)C2 c1(C(=O)NC2CC(N(C(c3nc(C)[nH]n3)=O)C)C2)ccc(-n2ccnc2S)cc1 N1(C(Cc2nc(CC)sc2)=O)CCCCC1C1(NC(=O)OC(C)(C)C)CC1 CC(C)S(=O)(=O)C(C)C(=O)NCCN1CCN(C(=O)COC2CC2(F)F)CC1 C1(C2(NC(C34C(NC(=O)CCC=CC(C)C)C5CC3C4C5)=O)CC2)(OC)CCC1 C(=O)(C1CCCc2sccc21)N(CCOCCCNC(C(CC=C)C)=O)C c1(C(=O)NC2CC(CCNC(c3cc(C)oc3C)=O)C2)nc(C)n(C2CC2)c1C Cc1cccc2nc(N3CCOCC(NC(c4coc(Cl)c4)=O)C3)oc12 C1(C(=O)OC)(C(=O)NC2CC2CNC(C2CC(F)(F)C2)=O)CCCC1 c1(OC)nc(CO)ccc1-c1ccc(NC(c2cncc(Cl)c2)=O)cc1 c1(C(N2CCC(O)(C(C)NC(CCCOCC)=O)C2)=O)cnc(C)c(N)c1 c1(C(=O)NCC(C)N(C)C(C2(C)CCN(C)CC2)=O)ccc2cccc(O)c2c1 CC12CC(C(N3CCN(C(=O)CC4C=CS(=O)(=O)C4)C(CO)C3)=O)(C1)C1(CO1)C2 c1(-c2onc(Cc3c(OC)ncc(Br)n3)n2)cnc2c(F)c(F)ccc2c1 C(CCCCCN=c1cc(C)nc(N2CC3CCC(C2)N3C)[nH]1)OC Cc1nn(C)c2c(N3CCC(NCCN(C)C)C3)nc(=NCCOCCO)[nH]c12 CCCC(C)(CC)C(=O)NCCCC(O)C(=O)NCCCCSC CC1=C(C(=O)NC2CCCC23CN(C(=O)C(C)=CC2CC2)C3)CCCO1 c1(C(=O)NC2C(OC)CN(C(CC3CCC(CC)CC3)=O)C2)cc(N)cc(O)n1 c1(N2C(C(=O)NC(C)(C)C3(SC)CC3)CC3(CC3)C2)nc(C)nc(Cl)c1COC C1(CC)(NC(=O)C(=O)NCC23CC(CO)(CO2)C3)CC(C)(C)C1 N1(C(C2CCCN(C(C)C)C2)=O)CC2OCCN(CC3(c4cc[nH]n4)CC3)C2C1 C1(NC(C(C(C)C)NC=O)=O)CCCN(C(=O)CC2COCCOC2)C1C c1(CC(C(=O)NC(C(OC)OC)C)C)ccc(O)c(O)c1 C(=O)(C(C)C(=O)NCc1nocc1C(=O)NCC(O)C(C)O)OC C1(NC(c2ccc(CNC(CN3CCC(=O)CC3)=O)nc2)=O)(CO)CC2CCCC12 Cc1c(C(=O)N(CCCN(C)C(c2ccnc(S)c2)=O)C)cnn1CCN(C)C C1(NC(c2c(CC)onc2C)=O)CN(C(=O)COC(F)F)CC2(CCC2)C1 C1(NC(CCc2ccn(C)n2)=O)CCCC12CN(C(=O)Cn1cnc(=N)[nH]1)C2 N#Cc1ccc(CC(N2CCCC(CNC(C3CCC(C(F)(F)F)O3)=O)C2)=O)cn1 c1(C(N2CCC(N(C(c3cnc(O)o3)=O)CC)C2)=O)cncc(Cl)c1 O=C(C1CCCc2c[nH]nc21)NCC12CCC(CC1)N2C(C1CC2C=CC1O2)=O CCC(Cc1ccccc1C)C(=O)NCC1CCN1C(c1ccccc1)=O c1(OC)ccc(-n2nnnc2N(C2CCOC2=O)CC(C)CO)cc1 c1(C(=O)NCC2(F)CN(C(C3(CCCC)CC3)=O)C2)csc2c(F)cccc12 C(C(C)N=c1[nH]c2c(c(=NCC(CO)C(C)(C)C)[nH]1)COCC2)c1ccc(C)s1 Cc1cc(C(=O)NCCC(C)N(C(=O)Cc2cnccn2)C)cc(Br)c1 c1(C(N2CCN(C(COCCC=C)=O)CC2COC)=O)cccn2cc(C)nc12 C(=O)(CCN=C(NCCC(F)F)NCC1CCCC(C)(C)C1)N(C)C C1(C(=O)NCC(C)(C)NC(c2csc(-c3ncccn3)n2)=O)CC2C=CC1C2 C=CC1(NC(N2CCC(Cc3ccccc3CC#N)C(C)C2)=O)CCCCC1 C(=O)(C(C#N)C1CC1)NCCCN(C(C)C)C(C1(c2ccccc2)CC1(F)F)=O C(=O)(CC(C(F)(F)F)NC(=O)C=CC1CCCN1C)N(C(C#C)C1CCC1)C NS(=O)(=O)CC(=O)N1CCCCC1NC(=O)COCC(F)(F)F c1(C(=O)NC2C3(CC(NC(Cc4cccc(C)c4)=O)C3)C2)c(O)nnc(C)c1C c1(OCC)ccc(Cl)cc1C(N1CC2(C1)CN(C(c1ccc(O)c(C)c1)=O)C2)=O CCS(=O)(=O)CC(=O)NC1CC=C(C(=O)NCc2ccc(F)cc2F)C1 Cc1nc(O)[nH]c1C(=O)NC(C1CCCCN1C(=O)CCc1cc(C)n(C)n1)C Cc1cc(C)n(-c2ccnc(N(CCO)C(=O)NC(C)Cc3cnccn3)n2)n1 c1(NC2(CNC(c3scc(OC)c3)=O)CCCC2)ncc(Cl)cc1[N+](=O)[O-] CC(C)C(C)C(C)CC(=O)NC1(CO)CCN(C(c2ccn(O)c(=O)c2)=O)CC1 CC(C)C(C)C(CNC(=O)CN1CCN(C)CC1)NC(=O)CCF Cc1ccc2c(c1)SC(C(=O)NCC(C)CNC(C1CCCC13CC3)=O)C2 N1(C(c2c(C)nco2)=O)CCC2(CCCN2C(=O)CC2CCC(C#N)C2)CC1 C(CC#CC)(C(=O)NCC1CCN(C2CC2)C1)NC(C1(C=C)CCC1)=O N1(C(c2c(C)nc(COC)s2)=O)CCCC(C)C1CNC(=O)Cc1ccsc1 C1(C(=O)NCCCOCCNC(C(=O)NC)=O)Cc2cccc(C)c2O1 [N-]=[N+]=NC1COCC1NC(=O)C(Cc1ccco1)NC(=O)CN=[N+]=[N-] c1(CNCC23C(CN(C(c4c(OC)nccc4)=O)C2)C3)cc(Br)ccc1Br CC(F)(F)C(F)C(=O)N(CCCNC(C1(C)CCNC1=O)=O)CCO C1(NC(COCCC(C)C)=O)CCCC(CNC(=O)CC2CC3(CC3)C2)C1 C1(C(=O)OCC)CCCCS1(=O)=O.n12cc(nn1)COCC=CCNC(=O)C2 c1(NC2CN(C(CCC(=O)Nc3nccs3)=O)C2)c(Br)cc(F)c(F)c1F CC(C)CCCC(C)CNC(=O)CC1C2CCCC2N1C(=O)C(C)OCOC N1(C(c2cn(CCC)nc2)=O)CC(C)OC2(CCN(C(=O)CC)CC2)C1 c1(NC(C(CC2CCOCC2)NC(c2ccc(O)nn2)=O)=O)ccc(F)cc1O Cc1ccc2c(c1)c(CCN(C(C)Cc1cccc(Cl)c1)C1CC1)cn2C C(=O)(C1CCCc2nn(C)cc21)N1CC2CCN(C(C(CC)CC)=O)C2C1 C1(CNC(c2c(C)ccc(C)c2)=O)CN(C(c2nscc2C)=O)CC(C)(C)C1 C1(=CC(=O)NCC2CC(NC(c3nncn3C3CC3)=O)C2)CN2CCC1CC2 C(=O)(CC(C1CC1)NC(=O)C(C)NC(C)=O)N(C(CC)CC)C O=C(CCC(=O)c1cccc(F)c1)NC1CC(CNC(C23CCC(CC2)O3)=O)C1 N1(C(c2ccc(C)cc2)=O)CCCC(C(=O)NCCC2NC(=O)NC2=O)CC1 CC1(C(=O)NCCCCC2CC2C)CC(O)CN1C(C1CC1(C)C(F)F)=O Cc1c(C(N2CCC2Cn2cc(CCc3nn[nH]n3)nn2)=O)sc2cncn12 CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NCC1(NC(C2(Cl)CC23CCC3)=O)CC1 n1(CC(=O)NCC2C(NC(CCCC#C)=O)C2)cnc2c1CCCC2 CCCC(C)(C)C(=O)NC1CC2(C1)CC2NC(=O)CCC(C)(C)OC CCCCCCC(CC)C(=O)N(CCNC(c1cnc(C)n1C)=O)CC1CC1 C12(C(=O)NCC3(F)CC(NC(c4cnc(O)c(F)c4)=O)C3)CCCC1C2(F)F C1(C(=O)NOCCCO)(CC=C)CC=CC1.C12CCC(C1)C(=O)N2C1CC1 CC1=NOC(C)(C(N2CC(CNC(=O)CC3C=NN(C)C3=O)C(O)C2)=O)C1 C1(CNC(c2c(CCC)nns2)=O)(CNC(=O)CC2CCOC2=O)CCCCC1 N1(C(C=Cc2c(C)ccnc2)=O)CCCC12CCN(C(C1(F)CCOC1)=O)CC2 c1(OC)ccc(=NC(=O)C2CC(F)CN(C(=O)C(C)SC)C2)[nH]n1 CCCCC(C(=O)N(CC(N1CC(C)OCC1C)=O)CC1CC1)C(C)C c1(C(=O)NC(CC)(C)CNC(c2ccc(C3CC3)cn2)=O)cc(O)nc(OC)n1 c1(CC(=O)NCCC2CN(C(C3(OC)CC3)=O)C2)csc2ccc(C)cc12 CCCCC(C)C(=O)NCCN(CC(C)O)C(C1CN(S(N)(=O)=O)C1)=O C1(C(=O)NCC(CNC(c2c(COC)cc[nH]2)=O)(C)F)CC2CC(=O)C1C2 c1(C(=O)NCC23C(CN(C(C4(CC)CC4)=O)C2)C3)cnc2[nH]cncc1-2 c1(NC2CC(OC)C2)cc(C(N2CCCC2CN=[N+]=[N-])=O)ncn1 C1(CNC(Cc2cncc(C)c2)=O)CN(C(c2cncc(N)c2)=O)CCN1C C(=O)(CCCN=[N+]=[N-])N1CCC(CNC(CCCn2c(C)ncc2)=O)C1 c1(C(=O)OCC)nn(C)cc1C(N1CCC(NC(=O)C(C)(F)F)C1)=O C(C(=O)CCN=c1cc(F)nc[nH]1)c1ccc(OCCC)cc1 c1(C(=O)NC2CN(C(COC)=O)CC2CC2CC2)nn2cccnc2c1Cl CCC(CC)(CO)C(=O)N1CCC(O)(C(C)NC(=O)CCCN(C)C(C)=O)C1 CCC(C)(C(=O)NCC1(F)CN(C(=O)C#CC2CCOC2)C1)C(N)=O c1(OC)cc(CC(=O)NC(CO)C(C)NC(C2CCC2)=O)ccc1C c1(N(C)C)cccc(C(N)=O)c1.c12ccc(cc1)NC(=O)NC21CC1 CC1(C)C2CCC(C(N3CC(F)CC3CNC(C3CCCO3)=O)=O)C1C2 N1(C(Cc2nc(C)sc2C)=O)CCC2CN(Cc3cnc(Cl)c(C)c3)CC12 CC1(C)CC(C(=O)NC2(C3CN(C(=O)CC4C=CCC4)C3)CC2)CC(C)(C)O1 C=C(C)CCCC(=O)NCC1COCCN(C(C2CSC2)=O)C1 c1(OC)ccc(F)c(C(=O)NCc2c(C)noc2C)c1.C12(CC(C)(C)C1)C(=O)N2 c1(OC)cccc(SCC(=O)NC2CC(COCCNC(=O)CN(C)C3CC3)C2)c1 C(CCN=c1cc(C)c(S(=O)(=O)Nc2cn(C)nc2OC)c[nH]1)NCC=C CCC(O)C(F)(F)C(=O)N1CC(c2cnnn2C)(N(C)C)C1 c1(-c2nnc(N(C)CC3(N)CCC(C)C3)n2C)cc(F)cc(Br)c1Cl c1(NC)cccc2[nH]ncc12.c12ccc(cc1)C(=O)N1CCCC1(C)C(=O)N2C1CC1 Cc1cc(O)c(C(=O)N(CCCCNC(=O)CCP(C)(C)=O)C)cc1Br C1(NC(c2nc(C)sc2C)=O)CCS(=O)(=O)C12CN(c1ncnc(Cl)c1C#N)C2 c1(C(N2C(C(=O)NC(C3C(C(=O)OC)C3)C)CCC2)=O)coc2c1COC2 C1(N(C(CC(C)C)=O)C)CN(C(=O)C(C)COc2ccccc2)CC1(C)C CC1CC(C(=O)NC(C)CC2CN(C(=O)C=C3CCN(C)C3)C2)CC(C)(C)C1 N1(C(C=CC(=O)OCC(C)C)=O)CCN(C(=O)C(C)(F)F)C(C)C1 CC1CC(NC(c2snnc2C2CC2)=O)CN(C(=O)CCn2cncn2)C1 S(=O)(=O)(c1cccnc1)NC1CCC(NC(=O)CCSc2ccccn2)C1 CCCCC(C(=O)NCCCC1(NC(c2cocc2C)=O)CC1)C(C)C C(C)(C(C)(C)NC(=O)CSC(F)F)NC(CCN(CCC)C)=O C(=O)(C(C)(C)C(C)(C)O)Nn1ccc(=NC(=O)C2(C(C)NCC3CC3)CC2)[nH]1 N1(C(CNC(C(CC)C)=O)=O)CCCC(N(C(=O)C2=CCCCC2)C)CC1 c1(C(=O)NC2(CNC(C=Cc3n(C)cnc3)=O)CC2)ccc2nc(CO)[nH]c2c1 CC1=C(C(=O)N2CCCC(CCNC(C3C4CC5C(C4=O)C35)=O)C2)CCC1 c1(NC(C)=O)ccc(C)c(C(=O)NCCC(C)NC(=O)C(F)C(F)(F)F)c1 N1(C(C=C(COC)C)=O)CC(CN(C)C(C2CCCCN2C)=O)C2(CC2)C1 NS(=O)(=O)CCCCCC(=O)NCCCCNC(=O)Cc1ccnc(Cl)c1F N1(C(Cc2c(C)ccs2)=O)CC2(CC(NC(C3(C)CCC(=O)NC3)=O)C2)C1 c1(CCNC(CCNc2c(O)ccc(C(C)=O)c2)=O)nc2c(o1)CCSC2 C1(C(N2C(C)CN(C(=O)C3=C(Cl)CC3)CC2)=O)CSC2(C)CCC(=O)N12 c1(C(=O)OC)cc(C(N2CCC(C)(NC(=O)COCC(F)F)C2)=O)c(C)o1 N1(C(C2CC(C)(C)O2)=O)CCCC2CN(C(=O)Nc3cc(Cl)cc(Cl)c3)CCC12 C1(NC(C(C)SC)=O)C2CC3C(C2)C13C(=O)N(C)CC1CCCC1(C)C CCC(CC(F)F)C(=O)N1CC(CNC(=O)CNC(N2CCCC2)=O)C(F)(F)C1 N1(C(C(CC)(C)C#N)=O)CCC2(CC1)CC(C)N(C(c1ccc(F)c(Cl)c1)=O)C2 N1(C(c2ccc(Cl)s2)C(=O)NCCC2(C)CC2)CCOCC1CC(N)=O C(=O)(CCCCC#N)NC(COC)OC(=O)C(=O)OC N1(C(c2cccc(COC(C)(C)C)c2)=O)CC2CC(F)(NC(N)=O)CC2C1 c1(C(N(CC(C)O)CCNC(COCC=C)=O)=O)cc2scnc2[nH]1 C(CC(C)(C)C(=O)N1CCC(O)C1)NC(C1(C(=O)OCC)CC1)=O Cc1nc(C(=O)NCC2CCN2C(=O)CC2CCOC2)c(C)n1C1CC1 c1(C(=O)NCc2cn(CC(CC)O)nn2)ccc2[nH]ccc2c1F N1(C(C(C)Oc2ccccc2)=O)CC2CCCCC2(NC(=O)C2=CCOC2)C1 CC#CCCCCNC(C12CC(NC(c3cc(C)[nH]c3C)=O)(C1)C2)=O N1(C(c2ccc(C#N)nc2)=O)CCC2CC2(NC(=O)CCCN2CCCC2)CC1 CCCCC(=O)C(=O)NC1CCC(CCC(=O)NCc2cccc(O)n2)C1 C1(NC(=O)CCc2cccnc2)C2CC(CN(C(=O)CCC3CCC3)C2)C1CO C1(NC(c2c(C)c[nH]c2)=O)CCCC(C(N2CC(CC(F)F)C2)=O)CC1 C1(F)(C(=O)NCCCC2N(C(=O)OC(C)(C)C)CCC2)C2CCCC12 C(=O)(C(CC)C(=O)N1CCC1(C)C(=O)OC)OCC.C12C=CCCC1C(=O)N2 C(=O)(C1=CCCC1P(C)(C)=O)N(CCN(C(c1c(CC)nccn1)=O)C(C)C)C C123CC(C4CC(=C)C4)(C1)C1(CN(C1)C(=O)NC2)O3.C12(C(=O)O)CC(C(=O)C3CC3)(CO1)C2.C1CC1.OC C1(CNC(C2C(OC)C2)=O)CN(C(=O)CCn2cnnn2)CC2(CCC2)O1 C1(NC(c2cccc(Br)c2)=O)CC2(CCC(NC(C3CC(O)C3)=O)CC2)C1 CC1OCCN(C(c2cc(C#N)cn2C)=O)C1C(=O)NCCC(C)(C)N(C)C C1(NC(c2[nH]cc(C)c2C)=O)CN(C(c2coc(Br)c2)=O)CCC1F C(=O)(C(C)(C)C(C)(C)C)N1CC(N(C(=O)C(c2cccc(Cl)c2)O)C)C1 n1(CC2CN(C(c3cncc(OC(F)F)c3)=O)C2)ccc2ccccc12 N1(C(CCN(CC#C)C(c2ncc(C)cc2C)=O)=O)CC(C)SC(C)C1 C(=O)(C1=NOC2COCC12)NCCN(C(=O)C#CC1CCCCC1)C(C)C C1(C(N2CCC(C)(O)C2)=O)CC2CC1CC2NC(c1ccccc1O)=O CCCCC(CC)CC(=O)NCCC(C)(C)C(=O)NCc1coc(C)c1 c1(C(=O)NCC(=C)CCNC(=O)CN2CCS(=O)CC2)ccc(=O)n(CCF)n1 C12(C(=O)OCC(=O)Nc3scc(C(C)(F)F)n3)COC(CF)(C1)C2 c1(C(C)NC(=O)CN(C)C(C2CC2)C2CC2)nncn1C n1(CC(=O)NCC2N(C(C(C)OC)=O)CCOC2)cnc2c(cnn2C)c1=O C1(NC(C23N(C(COCCC#C)=O)CC(C)(C2)C3)=O)CCc2nn[nH]c2C1 Cc1c(C(=O)NCC#CCNC(c2cc(O)n(C)n2)=O)nnn1C Cc1cc(Cl)c(C)c(C(=O)NCC2CCN(C(=O)CCc3cscn3)C2)c1N C1(C(=O)Nc2cccc(NC=O)c2)(NC(c2c(C)nccn2)=O)CCC(C)(C)C1 CS(=O)C1CN(S(=O)(=O)CC2CC2Cl)C1 Cc1cc(C)nc(SCC(N2CCC(NC(c3cscc3C(F)F)=O)C2C)=O)n1 Cc1ccc(C(N2CCCC(O)(CNC(=O)CC3CCCCO3)C2)=O)cc1O c1(CN(C2CN(C(c3cc(Cl)cnc3Cl)=O)C2)C)ccn2ccnc2c1 c1(C(=O)NC(C2CN(C(C3(C(F)(F)F)CC(=C)C3)=O)C2)C)nc(O)nc(O)c1F C(CC(C(C)(C)C)NC(c1cn2ccsc2n1)=O)N(C)C(c1csc(Cl)n1)=O C(C(C)C)(C(O)C(=O)NCC1CCN(C(c2coc(C(C)C)n2)=O)C12CC2)OC c1(C(=O)NC(C2CN(C(C3(C=C)CCC3)=O)C2)C)csc2cc(Cl)cnc12 c1(C(=O)NCC(=O)NCC2CCC(NC(C3COC(=O)C3)=O)C2)cccc(F)c1 C1(CC)CCCC1(C)C(=O)NCCN(C(c1ccc(SC)o1)=O)CC1CC1.C(C)(=O)N CCC(CC)(CO)C(=O)NC1CCC(CNC(=O)C2=NNC(=O)C2)C1 N1(C(C2=C(C)OCC2)=O)CCCC1C1CCCN1C(C1C2CCC1CC2)=O c1(C(C(N2CC(NC(COCCOCC)=O)C(C)C2)=O)C)ccc(F)cc1F c1(-c2cnc(CNCc3cc(O)cc(Cl)c3)nc2)ccc(F)c(O)c1F N1(C(C(c2c(C)nn(C)c2)O)=O)CCC(NC(=O)CN2CCN(C)CC2)C1(C)C C1(NC(Cc2cccc(CC)c2)=O)CCN(C(C2CCCC(F)(F)C2)=O)C12CC2 C(=O)(C(C#N)C(C)(C)C)NC(CNC(Cc1nnc(C)s1)=O)(C)CC(C)C c1(C(=O)NCC2(C)CCC(NC(C(C)(C)Cc3cnn[nH]3)=O)C2)cc(Cl)nnc1O c1(CC(=O)NCCCC(C)NC(c2ccc(Cl)cc2)=O)ccc(S(N)(=O)=O)s1 N1(C(c2ccc(CC)c(Cl)c2)=O)CC2CC(NC(=O)CC(C)(C)OC)CC2C1 S(=O)(=O)(c1cccc(Cl)c1)NCC(=O)NCC1CCN(S(CC)(=O)=O)CC1 C12(C(N(C3CCCN(C(=O)C=Cc4cscn4)C3)CC)=O)CCCC1C2(F)F c1(SC)ccc(C(=O)NC2(C3CCCN3C(=O)C=C(C)C(C)C)CC2)o1 C(=O)(CCC(=O)NCCC1(NC(=O)CN(C2CCS(=O)(=O)C2)C)CC1)NCC C(=O)(C(C)Cn1ccc(C)n1)NCCN(C(=O)C(n1ccc(C(F)F)n1)C)CC N1(C(C(C)CO)=O)CCN(C(=O)C2=COCCC2)CC1c1ccncc1 c1(C(=O)NC(C)COC(=O)Cc2ccc(F)cc2)ncc(Br)cc1N c1(NCC(CNC(=O)Cc2cccnc2)O)nc2ncc(Cl)cc2s1 N1(c2nc(=N)[nH]cc2)CCCC(C2(NC(c3nc(Cl)c(Cl)s3)=O)CC2)C1 Cc1c(C(=O)NC(C(N2CCOCC2(C)C)=O)C2CC2)cccc1O CC1CC(NC(=O)CNc2ccccc2)CN1S(=O)(=O)CC1CC1 C(=O)(CCC1=NNC(=O)CC1)NCC1(CNC(c2ccc(CC)c(Cl)c2)=O)CC1 O=C1CCN(CC(N2CCC(CCCNC(c3cnsc3)=O)CC2)=O)CC1 N1(C(C(CC)O)=O)CCN(C(CNC(c2ocnc2C2CC2)=O)C(F)(F)F)CC1 C(=O)(C(CNC(c1coc(C(C)C)n1)=O)C(C)C)NCc1c(CC)cncc1 C1(CNC(c2c(C)snc2)=O)COCCN(C(C2CC(C3CC3)=NO2)=O)C1 c1(CC)ccc(OCC(=O)NC(C)(CNC(=O)CC2CC3CC3C2)C(C)C)cc1 c1(NC2(CO)CCCN(C(C3N(C)CCCC3)=O)C2)ncnn2c(Br)ccc12 C1(n2cc(CCN(C(C)=O)C(CC(C)(C)C)C)nn2)CCC(C(C)(O)CBr)CC1 C1(C(=O)NC2CCCCC2CC(N2C3CCC(C3)C2CO)=O)CC12CCOCC2 c1(CNC(=O)COC2CCCC2C2CC2)ccc(S(=O)(=O)N2CCOCC2)s1 C(=O)(C#CC(C)(C)C)NC1C(NC(CCc2scc(C)n2)=O)CC1 C1(CNC(c2c(C)nn(C)c2)=O)CN(C(=O)CC2CCCCO2)C2CCCC2O1 N1(C(CCC(=O)OCC)=O)CCCCC(NC(c2ccc(CSC)o2)=O)C1 c1(CC(N2CC(CC(C)NC(c3cc(O)ncc3F)=O)C2)=O)ccc(F)c(F)c1 Cc1cc(C)c(C(=O)NCCN(C)C(C2(C)CCCCC2(F)F)=O)c(S)n1 c1(CCC)ccc(C(N2CC(NC(c3cnnn3C3CC3)=O)C2)=O)s1 C1(NC(c2cccc(C#C)c2)=O)CCN(C(=O)CS(=O)(=O)NC(C)C)C12CCC2 C(=O)(CCC1=CCCCC1)N1C(CO)CC(NC(C2CN3CCCC2C3)=O)C1 C1(C)(C(N2CCC(O)(CCNC(C3C(C)C3)=O)C2)=O)CCS(=O)(=O)CC1 N1(C(c2nccc(OC)c2)=O)CCC(O)CC1C(=O)NCC(C)CC1CCCC1 C1(NC(CNC(C(C)C)=O)=O)CC(C)(NC(=O)COCC2(F)CC2)C1 N1(C(c2ccc(C)cc2C)=O)CCC(C2CCCN(C(C3CCCC3O)=O)C2)C1 N1(n2cc(C3(F)CN(C(c4ncc(Cl)s4)=O)C3)nn2)CC2CCC1C(O)C2 c1(C(N2C3CC(NC(C(C)(C)F)=O)CC2CC3)=O)c[nH]c2cc([N+](=O)[O-])ccc12 N1(C(C(n2c(C)ncc2)C)=O)CCn2ncc(CNC(C3CC34CCC4)=O)c2C1 C(=O)(C(F)(CNC(=O)CNC(=O)NC1CC1)C(C)C)N1CCC(CC)C1=O C12(C(N3CCOC(CC4CC4)C3)=O)CCC(C(=O)NCC3(CO)CC3)(CC1)CC2 Cc1nn(CC(=O)NC2CCCC2CNC(c2cc(O)cc(Cl)c2)=O)c(C)c1Cl Cc1ccc(C=CC(=O)NC2CCN(C(C3CC3C(F)(F)F)=O)C2C(C)C)o1 C1(C(F)(F)F)(C(=O)NC(c2ccc(F)cc2)c2ccncn2)OC2CCC1CC2 c1(CNC(C(C2(C)CC2)NC(C(COC)OC)=O)=O)cncc(F)c1 c1(C(=O)NC(C2OCCN(c3snc(COC)n3)C2)C)coc2c1CCCC2 C(N=c1nc(CC2CC2)[nH]s1)C1CCC(C(C(C(C)C)n2cnnc2)=O)C1 C=CCC(CNC(C1C=CCC1)=O)C(=O)NC(C)(C=C)CC C(=O)(CCCCCC(C)O)N1CC(OC)(CNC(C2CC23CC(O)C3)=O)C1 c1(OCC=C)cc(Br)ccc1C(N1CC2CCC2(CC(=O)N(C)C)C1)=O C1(SC)CN(C(=O)CC2(C)CC2(Cl)Cl)CC1NC(C1(n2cccn2)CCC1)=O C(=O)(C#CC(C)(C)C)N1CCCC(N(C(C(C(C)C)C)=O)C)C1 C1(CN(C(=O)COCC2CC2)C)CC2CCC(C1)N2C(c1cc(O)cc(O)n1)=O N1(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)C2)CCC(S)c2cc(F)ccc21 c1(CC)ncc(C(N2CC(F)CC2CNC(c2cc(C3CC3)on2)=O)=O)c(O)n1 C1(CNC(CC=CC=C)=O)COCCN(C(=O)C(C(C)(C)C)NC(C)=O)C1 N1(C(CC(C(C)C)(F)F)=O)C2CCC1CN(C(c1ccsn1)=O)CC2 C1(c2c(C)ncs2)CCN(c2ccnc(NC(c3ncccc3F)C)n2)CC1 N1(C(N2CCCC(C)C2)=O)CCC2(C1)CN(C(c1nc(O)nc(O)c1F)=O)C2 Cc1cc(Cl)cc(N(C(=O)C(c2ccc(Br)s2)C)CCO)c1I C(=O)(C1CCCn2ncnc21)N(CCC(C(C)C)Nc1cc(O)nc(O)n1)C c1(OC)ccc(SCC(=O)N(CC(C)O)CCNC(c2oncc2C)=O)cc1 C1(NC(Cc2n[nH]c(=N)s2)=O)CCCCC12CCN(C(C1CCC1)=O)CC2 C1(C2CCC2)(C(N2C(CNC(=O)C(c3ccc(F)cc3)=O)CC2)=O)CCC1 C1(C)(CNC(CN(C(C)C)C)=O)CN(C(=O)Cc2cn(C)cn2)C(C)(C)C1 N1(C(=O)Cc2ccnn2C2CC2(F)F)CC2CN(C(C3CCCC3)=O)CC2C1 Cc1ccnc(C)c1C(=O)NCC12CC(CO1)N(C(c1cc(Cl)c(C)cn1)=O)C2 N1(C(C(c2nccc(C)c2)(C)C)=O)CCCCC2(C1)CN(C(C1(C)CC1C)=O)C2 CC(C)CC(CNC(=O)CN1CC2CC2C1)NC(=O)COCCCF n1(CC)nc(C)c(C(=O)NCCCCCN(C)C(C2CCCOCC2)=O)c1Cl C(=O)(C(C)CCC(C)(C)C)N(CC(N1CC(OCC)C1)=O)CC1CC1 N1(CCC(=O)N(CC(C)NC(=O)CCc2ccccc2)CC)CCCCC1=O C1(C(=O)NCCOCCCC)CN(C(=O)CCc2ccc(N(C)C)[nH]2)CCCO1 CN=c1[nH]nc(CC(=O)NC2CN(C(=O)CCCOC(C)C)CC2C)s1 N1(C(c2n(OC)cnc2C)=O)CCC2(CC1)CC2CNC(C1(Br)CC1)=O C#Cc1ccc(OC)c(C(=O)NC(C2CCCN2C(c2ncccn2)=O)C)c1 N1(C(c2cccc(F)c2C(F)F)=O)CC2OCCN(C(=O)CC34CC(C3)C4)C2C1 C1(COC(CCC=C=C)=O)CCC(=O)N(C(=O)C=C2CCCCC2)CC1 C1(C(N(CC(CN(C)C(c2c[nH]nc2C2CCCO2)=O)O)C)=O)CC=CCC1 Cc1cnc(C(=O)NCC2CC2CNC(C2CCC2)=O)c(C)c1 C1(CC(=O)NC2COCC2n2cc(COCCOCCO)nn2)CC2CC2C1 CC(CNC(C1CC(NC(C2CC2NC(N)=O)=O)C1)=O)(CO)OCCCl c1(C(C(=O)NCC(C)CN(C)C(c2coc(O)n2)=O)C)ccc([N+](=O)[O-])cc1 N1(C(c2ccc(C)o2)=O)CCN(C(=O)Cc2cnn(CCF)c2)C(CF)C1 C1(C(N(CCC(c2cccs2)NC(=O)C2=CCSC2)C)=O)CCC2CC1CO2 N(C1c2ccccc2OCC1F)C(=O)NCc1ccc(OCCC)cc1 Cc1c(C(N2CCC(C(C)NC(C3(CO)CC3)=O)CC2)=O)ccn1C1CC1 N1(C(c2cc(CCC)n(C)n2)=O)C(CNC(=O)CCOC2CC2)CC2COCC12 c1(C(N2C(CNC(C(C=CC)O)=O)CC(O)C2)=O)cc(C)nc2c1CCCC2 C(CC)(CCCC(=O)NCC1(CN=[N+]=[N-])CC1)NC(c1ccc(C#C)cn1)=O c1(C(c2n(CC)nnn2)NCc2cc(C(=O)OC)cs2)c(F)cc(Cl)cc1F Cc1cc(C(=O)N(C)CCNC(c2cccnn2)=O)c2c(O)nn(C)c2n1 C12(C(=O)NC(C3CN(C(C4CC4[N+](=O)[O-])=O)CCO3)C)CC(C)(CO1)C2 c1(C(N2C(C)CC(CNC(C(CCCC)(C)F)=O)C2)=O)ccc(P(C)(C)=O)nc1 C1(CCC(=O)OC(C)(C)C)CN(C(c2ccccc2F)=O)CCO1 C1(C(=O)NC(CNC(c2cccnc2C(F)(F)F)=O)C(C)C)(OC)CCCOC1 C1(C(=O)NC(C(=O)NCC(C(C)C)CO)c2cn[nH]c2)CCC(C2CC2)C1 N1(C(C)(C)C)CC(O)CC1C(=O)NCc1[nH]ccc1-c1ccccc1 c1(OC)ccccc1C(C)=CC(=O)OC(c1cccc([N+](=O)[O-])c1)C C(=O)(C(O)CCNC(=O)CN1CCCC1C)NCCSc1onc(C)n1 CCCS(=O)(=O)C(C)C(=O)NCC1(O)CCN(C(c2cc(F)c(F)cc2Cl)=O)C1 c1(NC(CC2(C)CCN(C(=O)C#CC3CC3)C2)=O)cnc2ccnn2c1 CCCCCC(F)C(=O)N1CC=C(C(=O)N2CCOC(C)C2)CC1 N1(C(CC(CCC)O)=O)CCC2(C1)CN(C(c1c[nH]nc1-c1ccncc1)=O)C2 c1(C(=O)NCCN(C(CC(=C)C)=O)CC2CC2)cc(N(C)C)cc(Br)c1 N1(C(C(c2cc(CO)on2)COC)=O)CCCC(OC)CCC1.c1ncn(C)c1C N1(C(c2c(-c3ccccc3)nc(C)n2C)=O)CCC(CNC(=O)CO)C(C)(C)C1 C1(C(=O)NCC2(CNC(CCc3n(C)ccc3)=O)CC2)CCc2nnnn2C1 C1(CNC(C2(COC)CC2)=O)CC2CCC1N2C(=O)CCC1CCCC(=O)N1 C(=O)(C1CCCc2sc(=N)[nH]c21)NCC1CN(C(C(c2n(C)ccn2)(F)F)=O)C1 C1(C)(C(=O)NCCC(=O)OCC)CCN(C(c2ccc(C(=O)OC)nc2)=O)C1 N1(CC)CC(n2cc(CNC3CCCC3O)nn2)C(C)C1.c12ccsc1C(=O)N2 C#Cc1cnc(NC(C)CNC(c2c[nH]nc2C(C)(C)C)=O)nc1 C12(C(=O)NC(=O)NCC)CCOC(CNC(=O)C(=O)Nc3ccco3)(C1)C2 Cc1nc(NC2CCN(C(c3cc(Cl)n(C)n3)=O)C(C)C2)cc(Cl)n1 N1(C(CCC(C)(C)F)=O)CC2(CCCC2NC(c2cnc(S)[nH]2)=O)C1 c1(C(=O)NC(C)CNC(=O)CC2CCCCO2)c(Cl)ccc([N+](=O)[O-])c1Cl CCCCCS(=O)(=O)CC(=O)N1CCSCC1CCNC(C1(SC)CC1)=O C1(C(=O)NCC(C(=O)OCC)C)CCN(C(C23CCC(CC2)CO3)=O)C(C)(C)C1 C1(C(N(CCSC)CC)=O)N(C(=O)C(CSC)OC)CCC1(C)C c1(C(=O)NC2C(CC)CCN2C(c2ccnc(OC)n2)=O)ccc(O)c(F)c1 CC1(CNC(c2ncsc2C2CC2)=O)CCCN(C(C2OC3CCC2CC3)=O)C1 CCC(C)(O)CCNC(=O)CC(CC1CC1)NC(c1nnc(S)n1C)=O Cn1cc(C(N2CCCC2(C)C(=O)NCCC(Cl)(Cl)Cl)=O)ncc1=O c1(C(=O)NCC2C(NC(Cc3nnc(C)s3)=O)C2)cc(C)n(NC(N)=O)c1C c1(CN2CC(NC(c3c(C)cccc3O)=O)C2)cccc([N+](=O)[O-])c1F C12(NC(C(C)NC(C)=O)=O)CCOCC1CN(C(c1cccn1C1CC1)=O)C2 C=CC1COCCN1C(C1C2CC1N(C(C1CCN1C(C)(C)C)=O)C2)=O c1(C(N(C(CC)C2CC2)CC)=O)ccc(CNC(=O)C(C)O)cc1 N1(C(C(C)C2CCC2)=O)CC23CCCC2(C1)CN(C(=O)C=Cc1ccccc1)C3 c1(C(C(=O)N(CC(C)O)CCNC(=O)Cc2cc[nH]n2)C)ccc(Br)cc1 N1(C(CCC)=O)C2CCC1CN(C(=O)CCC=Cc1ccccc1)CC2 N1(C(c2nc(Br)cn2C)C(=O)NCCCSC)CCC(CO)(CO)CC1 C=CC(C)(C)CC(=O)NCC(C)(CNC(=O)C(F)C1CCC1)OC c1(N(C)C)ccc(CCC(=O)NC2CN(C(=O)CCc3cnco3)C2)cn1 c1(C(C)C)nnc(C=CC(=O)NCCC(C)NC(=O)CC2CC2(Cl)Cl)o1 C(CC(F)F)(C(=O)NCC1(O)CC(O)C1)N(C(=O)CCC1CCOCC1)C C=C=CC(C)C(=O)N1CCC(C(=O)NCCN2CCC(OC)C2)(OC)C1 N1(C(c2cnnn2C)C(=O)NCc2cccc(OC)c2)CCC2(CC1)OCCO2 C1(NC(CC(=O)OCC)=O)CC2CN(C(=O)C(C)CSC)CC2C1 C(=O)(C(C)(C)CC(=O)NC1(CCNC(=O)C(C)(C)c2cc[nH]n2)CCCC1)OC N12CC3(CC3)CC1C2=O.c1(NC(C2C3COCC23)=O)ccccc1-c1ccco1 c1(C(=O)NC(c2c(C(=O)NC(C)CC3CCOCC3)con2)C)cc[n+]([O-])cc1 C1(C(N2CCOCC(CNC(CCCOC(C)C)=O)C2)=O)CC2(CCCCC2)C1 C#Cc1ccc(C(=O)NC2(CNC(c3n[nH]c(C)n3)=O)CCCC2)cc1Cl c1(C(=O)NC2CC(F)(CNC(c3ccnn3CCF)=O)C2)cc2c(o1)CCCC2 c1(C(=O)NCc2c(C(N(CC=C)CC)=O)occ2)cnn2c1OCC2 C1(C(=O)OC)CC12CCCN(C(c1c(Cl)ccc(Cl)c1OC)=O)C2 N1(C(c2cc(C)sc2C)=O)CCCCC(C(N2CCC(OCCF)C2)=O)C1 C#Cc1cccc(C(N2CC(NC(C3(C)CC(O)CN3C)=O)CC(C)C2)=O)c1Cl C1(CC(=O)N(C)CC2(O)CC2)CCCC(NC(c2cccc(C3CC3)c2)=O)C1 N1(C(C(C)OCC2CC2)=O)CCC2(CCN(c3nc(C4CC4)ns3)C2)C1 c1(COC)ccc(C(N2CCCC(CNC(c3ccc(OC)nn3)=O)C2)=O)cc1 C1(C(=O)OC)(C(=O)NC2CC2CNC(c2cc(C3CC3)cs2)=O)CC=CC1 c1(C(N2CC(NC(c3ccc(C)c(CO)c3)=O)C(C)C2)=O)nc2ccccc2s1 C12(C(=O)NCC(CC#C)(C)C)CCN(C(c3csc(CO)n3)=O)CCC1C2 N1(C(CCN(CC(F)(F)F)C)=O)CC2CCC1CN2C(c1cnc[nH]1)=O Cc1cc(=O)c(C(=O)NCCC2CCN(C(C3CCC3(C)C)=O)C2)cn1C1CC1 N1(C(C2C(NC(c3cc(C(N)=O)[nH]n3)=O)CCO2)=O)C2C=CCC1CCC2 c1(CC)ncoc1C(N1CCC1CC(=O)N(CC)Cc1ccccn1)=O C(=O)(CC(C)(C)C(=O)NCC12CCCC1N(C(C1CC(O)C1)=O)CC2)OC N1(C(C2(C)COC2)=O)CC(NC(C2(O)CCSC2)=O)C(C(F)F)C1 C1(NC(C2CCc3nncn3C2)=O)CC2(CCCN(C(c3cnc(Cl)s3)=O)C2)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCC2CCCC(C1)N2C(c1cn(C)cn1)=O c1(NC(C2CCN(C(C3CCc4nc[nH]c4C3)=O)C2)=O)ccc2cnccc2c1 CC1(C)C(CNC(c2coc(C3CCCCC3)n2)=O)CCN1C(c1ccsc1)=O CCCC(CC)CCC(=O)N1CC2CC2C1C(=O)NCC1(O)CCC(C)(C)C1 c12ccc3c(c1)CCCC3NC(=O)C(=O)N2.CCCC(C1CC1)OC.C1(=O)CO1 CC1(CNC(c2cnoc2)=O)CCCN(C(=O)Cc2csc(C(F)(F)F)n2)C1 N1(C(C(C)=CC)=O)C2CCC1CC(CNC(c1cccc(C(N)=O)n1)=O)C2 c1(NCC(C)(C)C(F)F)ccc(S(=O)(=O)N2CCOC3COCC3C2)cc1Br C(=O)(C(O)C(F)(F)F)NC(C1CCN(C(C(C2CCOCC2)C)=O)CC1)CO c1(CC(C)NC(=O)Nc2ccc(-n3cnnn3)cc2)cccc(F)c1 C1(NC(Cc2nc(C)oc2)=O)CCCC(NC(c2ncccc2NC2CC2)=O)C1 C1(N(C(c2scc(C)c2)=O)CC2CC2)CCN(C(c2ccnn2CCF)=O)CC1 N1(C(Cc2c(C)scc2)=O)CCC(C(C)CNC(=O)CC2CCNC2=O)CC1 c1(C(=O)NCC2N(Cc3ccnc(SC)n3)CC2)cc2ncccc2s1 C1(NC(C(C2CCCC2)SCC)=O)CCCCC1CNC(c1nc(Cl)cs1)=O CC(CC(=O)NCC1CN(C(=O)C(C)(C)F)CCO1)C(F)(F)F c1(C(=O)OCC(c2ccc(C(CC)C)cc2)=O)cc(=O)n(C)cc1Br C1(CNC(CC(=O)OC)=O)CN(C(c2coc(S(=O)(=O)NC)c2)=O)CC(C)(C)C1 CN1CC(=O)OCC1C(N1CC(O)CC1CNC(C1CC(C)(O)C1)=O)=O C(=O)(C1c2c[nH]nc2CCC1C)N(CCNC(CCC=C)=O)CC1CC1 c1(C(CNC(=O)CC2CN(C)C2)NC(C2(CC)CCC2)=O)ccc(C)cc1 C1(NC(=O)CN2CSCC2=O)COC2(C1)CN(C(c1cn(CCCF)nn1)=O)C2 c1(C(N2CCC(COC)(CNC(=O)CNC=O)C2)=O)c(Cl)nc2sc(C)cn12 C1(CNC(=O)Cc2cnoc2)CN(C(C2CC(n3ccnn3)C2)=O)CC1(F)CO N1(C(C(C)C2CC2)=O)CC(CNC(C2(CF)CCOCC2)=O)OC(C(F)(F)F)C1 N1(C(c2c(CNC(c3ccc(CC)nc3)=O)c[nH]n2)=O)CCCC12CCNC2=O c1(C(N2CC(NCc3cn(C)nc3)C2)=O)cc([N+](=O)[O-])c(Cl)c([N+](=O)[O-])c1 c1(C(N(C2CCN(C(C3CCCCS3)=O)C2)C)=O)ccc(C#N)o1 N1(C(c2ccc(F)c(C)c2O)=O)CCN(C(C2CCN(C)C2C)=O)CC(C)(F)C1 Cn1c(C(=O)NC2CCCCC2NC(=O)C(c2cccnc2)O)cnc1O C1(C(=O)NCCCN(CCO)C(c2cnc(C3CC3)nc2)=O)CC2CCC(C1)C2 C(CC)(C(=O)NC(C1CCCCC1)CNC(c1cscc1OC)=O)OCC C(=O)(CCCCCF)N1CCCC(CC(=O)NCc2n[nH]c(C3CC3)n2)C1 c1(C(N2CCN(C(CCCCC)=O)C(c3cn[nH]c3)C2)=O)c(C)cc(F)cc1C c1(CC(=O)NCC(C2(O)CCN(C(c3c(C)ocn3)=O)C2)C)cccc(F)c1F C1(NC(C(C(CC)C)O)=O)CN(C(=O)C(C)C2CC2)CC12CCOCC2 C1(O)(Cn2cc(-c3ncc(C)o3)nn2)CCN(C(c2ccsc2Br)=O)C1 C=CCC(C)(CC=C)NC(C12CC(NC(=O)C(F)n3ccnc3)(C1)C2)=O c1(OC)cc(N)c(Cl)cc1C(N1CC(CNC(C2CC2C(F)F)=O)C(O)C1)=O c1(OC)cccc(Br)c1C(=O)NC(CNC(=O)C1=COCCO1)C(C)(C)C c1(CC)n[nH]c(=NCCC2CN(C(C3(C(=O)OC)CCCO3)=O)C2)s1 c1(OCC(=O)NCCCC(C)NC(C2(O)CCSC2)=O)cc(F)cc(F)c1 CC1CCC(CNC(=O)CC2CCN2C(N)=O)N(C(=O)C=Cc2cc[nH]n2)C1 CCCCC(C(=O)N1CC(CNC(=O)CN(C)C(=O)OC)C2(CC2)C1)N(C)C N1(C(C(CC)CCOC)=O)CC(NC(=O)Cc2cscn2)C2CCCCC12 N1(C(Cc2c(C)occ2)=O)CC(C)C(NC(=O)CCc2ccoc2)C(C)C1 Nc1ccc(S(=O)(=O)NC(c2cn3ccc(Br)cc3n2)=O)cc1Br C1(CN(C(=O)C(N)=O)C)CCCN(C(c2cc(-c3cccc(Cl)c3)on2)=O)C1 C1(NC(c2cncc(CNC(C(n3ccc(C)n3)C)=O)c2)=O)C(=O)NCC1(C)C C(=O)(C(C(C)(C)C)OC)NCC(CO)NC(c1cncc(CC)c1)=O N1(C(CC(CC)SC)=O)CCCCC(NC(c2ncccc2Cl)=O)C1 C1(NC(=O)COC2CC2(F)F)CCC2(CC1)CCN(C(=O)COCC1CC1)C2 C#CC1(C(=O)NCCN2CC3CC3C2)CCN(C(c2nnsc2N)=O)CC1 C#Cc1ccccc1CC(=O)NC1(C(=O)NCc2n[nH]c(C)n2)CCC(C)(C)C1 Cc1cc(=NC(CCF)C2CCCCC2)[nH]c(N2CCC(CS(C)(=O)=O)CC2)n1 C1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C(C)C)CCC2(CCC2)CC1 c1(C(N2CC3CC(C(N4C(C)(C(C)C)CC4)=O)(C2)C3)=O)nccc2[nH]ccc12 N1(C(c2c(C)[nH]cc2)=O)CCOC2(CCCN(C(C3CC(C(C)C)C3)=O)C2)C1 c1(N(CC(C)NC(C2CC(CC(C)C)OCC2)=O)C)nc2ccc(F)cc2o1 C1(C(N2CCCC2C2CCN(C(C3(F)CCC3)=O)C2)=O)Cc2cc(Cl)ccc2O1 C=CC(O)C(=O)NCCCN(CCCNC(c1coc(COC)n1)=O)C c1(OC)ccc(F)c(CNc2cccnc2C(=O)Nc2ccc(O)c(Cl)c2Cl)c1Br C1(C2(C)N=N2)CCCN(C(C2CCN2C(c2ccc(Cl)cc2)=O)=O)C1 c1(NC(C(COC)NC(=O)Cc2cncs2)=O)ccccc1CCO C1(C)(CNC(CCC2CCC(C)O2)=O)CCN(C(C2(F)CCOCC2)=O)CC1 N(C1CCc2cc(F)c(F)cc21)C(=O)NC1CCCC(C(=O)OC)C1 C=CC1COCCN1C(C1CCN(C(=O)CCC2CCCC2)C1)=O c1(CC(N2C(C)C(NC(=O)CCC3CC3)CC2)=O)cc2ccccc2nc1O c1(N2CCC(C)C(NC(c3cccc4ncoc34)=O)C2)ncnc(Cl)c1[N+](=O)[O-] N1(C(COc2c(C)cccc2)=O)CCC2(CCC2)C(CNC(=O)CCF)C1 c1(C(=O)NC(CC#C)C(=O)NCc2cnccc2Cl)cnn2ccc(Cl)c(F)c12 N1(C(C2CCC(C)C2)=O)CCC2(CC1)CCN(C(c1cnn3ccccc13)=O)C2 N1(C(c2c(C)ccc(O)c2)=O)CC(C)N(C(c2cc(C3CC3)ns2)=O)CC1C Cc1nnsc1C(=O)NCC1CC1CNC(C1(c2ccccc2)CC1(F)F)=O.C1(S)CC1 C1(CC)CCCN2C(=O)N(CCCCCC3CC3)C(=O)C2C1 Cc1cc2ncn(C)c2cc1C(N1CCCCC1(C)c1ccccc1)=O N1(C(C=CC)=O)CCC2CCN(C(c3ccc(C)s3)=O)C2C1 N1(C(CC)=O)CCN(C(C2CCCC(=O)N2C)=O)C(c2ccncc2)C1 C1(C)(CC)CC(C(=O)NCC2CN(C(=O)CCCF)CC2(C)C)CCO1 C(CC(C)C(=O)NCCOCCCN(C(=O)CSc1nccn1C)C)OC O=C1Cc2c(C(N3Cc4[nH]nc(C(N5CCC(F)(F)C5)=O)c4C3)=O)cccc2N1 CCC(C)CC(=O)NCC1CCCCN1C(=O)C=CCN1CCC1 C(=O)(C1=C(C)OCC1)C(=O)C=CCF.C(CC(=O)NCC1(N)CCC1)NC(C)=O c1(C(N2CCC(OC3CCOCC3)CC2)=O)ccccc1Sc1ccccc1 CC(c1ccccc1F)=CC(=O)NC(C)C(C)NC(=O)Cc1ccc(C)cc1 CCCC(CCC)C(=O)N1CC2C(NC(c3nc(Cl)ccc3F)=O)C2C1 c1(C(N2CCC(F)(CNC(CNCCC#C)=O)CC2)=O)c(C)cc(OC)cc1C C1(CNCc2ccccc2C(F)(F)F)COc2cscc2O1 CC1CNC(=O)CN1C(C1C=CCN1C(=O)CC(F)(F)F)=O C1(CNC(CCOC)=O)CC2(CO1)CN(C(=O)CCCC(OC)OC)C2 C(CCCCNC(=O)C(C)(C)c1ccns1)NC(CNC(=O)OC(C)(C)C)=O N1(C(Cc2c(C)ncs2)=O)CC(C)CN(C(C2CC3CCCCN3C2)=O)C(C)C1 C1(NC(COCCOC)=O)CN(C(c2cc(C3CCCN3C)[nH]n2)=O)CC(F)(F)C1 c1(C(=O)OC)ccc(C(=O)OCc2nnc(-c3ccc(C)cc3)n2C2CC2)n1C Cc1ccc(C#N)cc1C(N1C2CCC1CN(C(=O)CC(C)F)C2)=O c1(CC(=O)NC2CCCC(NC(C3(C)CCCOC3)=O)C2)ccccc1[N+](=O)[O-] N1(C(C2CC(CNC(c3c(C(N)=O)occ3)=O)OC2)=O)CCC2(CC1)N=N2 Cc1cc(=NC2CCC3CN(C(=O)C(C)(C)S(C)(=O)=O)CC3C2)[nH]cn1 C(C(=O)N(CCC)OC)N1CCCC(NC(C(CC=CCC)C)=O)CC1 C(=O)(C1=NNC(=O)CC1)N1CCC(N(C(=O)C2=CCCS2)CC)C1 CCC(CC)(CC)C(C(=O)N1CC(C(=O)OC)C(C)C1)OC O(NC(=O)C(COCC)C(C)C)CCCc1cccc2c[nH]nc12 Cn1nnc(C(=O)NCC(CO)NC(=O)CNc2ccccn2)c1N CC(C)CC(C)(CNC(c1cc(CO)[nH]n1)=O)NC(c1cc(Cl)cn1C)=O C(=O)(N1CCCc2ccnn21)C12CCCN1C2=O.C1(CC)CC2CC1CC2=O C12CCN(CC1)C(=O)C(CO)NC2C.C1(C(=O)NC(N)=O)CC1C(F)(F)F c1(CCC)n[nH]c(=NC2CN(C(c3cnc4n3CCCC4)=O)CC23CCC3)s1 n1(CC(=O)NC2CCC(N(C(=O)C(N)=O)C)C2)cnc2ccc(F)cc2c1=O C1(CNC(CCc2n(C)ccn2)=O)(CNC(C2CC(=C3CC3)C2)=O)CC12CCC2 C1(CNC(CC(C)C(C)(C)C)=O)(CO)CC12CCN(C(=O)Cc1cnc[nH]1)CC2 CC(C)C(C(=O)NCC1CCCN1C(C1CC(C)(O)C1)=O)NC(=O)C(C)(C)C C1(C(=O)NC2CN(C(C)C)CC2C)CCCCN(C(C2CC2C#N)=O)C1 CC(C)CC(C(=O)NCCNC(=O)Nc1cnn(C)c1)NC(=O)CC1(CO)CC1 CCCCS(=O)(=O)CC(=O)NCC1CC2CCC1N(C(=O)C1=CCSC1)C2 C1(N(C(=O)CCc2nc[nH]n2)CC)CCN(C(C2(C3CCCO3)CCC2)=O)CC1 C1(NC(C2C(C)C2)=O)Cc2ccccc2N(C(C2CCCN2C=O)=O)C1 c1(OC)ccc(F)cc1C(c1nnnn1C(C)C)NC(C)CCCOC CC1(c2cn(CC(N3CC(NC(=O)CCCn4cccc4)C3)=O)nn2)CCOC1 CCCC(CNC(=O)C(C)S(N)(=O)=O)C(=O)NC(c1ncccc1C)C c1(C(=O)O)ccc(CN2CCCCC2C(=O)NCCOCCC(F)(F)F)nc1 C1(CC)(NC(C23CCN(CC2)CC3)=O)CCCN(C(=O)CNc2ncccn2)C1 c1(OC)ccc(C(N2CCN(C(c3cnc(Cl)cc3Cl)=O)C(CO)C2)=O)nc1Cl c1(C(N2C(C)CC(NC(c3n[nH]cc3Cl)=O)C2)=O)cc2cc(Cl)ccn2n1 C1(CNC(C(CCC)O)=O)CN(C(=O)CCN2CCCS2(=O)=O)CCC1CO c1(C(=O)NC2CCC(CNC(=O)Cc3ccno3)C2)ccc2cccnn12 c1(C(=O)NCc2ccc(-c3cc[nH]n3)cc2F)cc(I)ccc1[N+](=O)[O-] C1(C)(C(=O)NCC(NOC)=O)CCCN(C(c2cc(C)n(C)c2C)=O)C1 CCCN(OC)C(=O)CC1CC=CCN1C(=O)CN1CCCCC1 C=CC(C)(CCOC)C(=O)NCCC(O)CNC(c1cnoc1C)=O c1(C(=O)NCC2CC(NC(c3ccccc3F)=O)C2)ccnc2ccc(F)nc12 c1(CC)cc(F)ccc1C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C c1(C(=O)OC)cc(C(=O)NC2CCCC2CNC(=O)CC2OCCO2)on1 c1(C(=O)NC(CN(C(=O)C(c2cncnc2)C)CC)C)cccc([N+](=O)[O-])c1N c1(C(CC(=O)NC2(C)CC(NC(c3nnc(C)s3)=O)C2)C)c(C)n[nH]c1C C(c1csc2ccccc12)=CC(N1C(CNC(C2CC(N(C)C)C2)=O)CCC1)=O c1(CNC(=O)Nc2nc(-c3nn[nH]n3)cs2)ccc(N2CCC(O)CC2)cc1 c1(OC)ccc(C(N2CC(NC(c3cc(C4CC4)on3)=O)CC(O)C2)=O)cc1C C(=O)(C(CC)C(=O)N1CCC1CC(N1CC2CC1CS2)=O)OCC CC1CC(CNC(c2cc(F)cs2)=O)CN1C(=O)COc1cccc(Br)c1 Cc1cccnc1CC(=O)NC(Cc1nccn1C)C(C)C Cc1cc(CC(=O)NC(C)C(=O)NCc2noc(C3CC3)n2)cs1 Cc1cc(C(=O)N(C2CN(C(c3ccon3)=O)CC2O)C)c(O)nn1 N1(CC(=O)NCCSC)CCN(C(=O)CCc2ccc(N(C)C)cc2)CC1 c1(C(=O)Nc2onc3ccccc23)ccc2c(C3=CCOCC3)n[nH]c2c1 c1(C(N(CC(C)CNC(=O)CC2(C)CCC2)C)=O)ccc(C(F)F)c(Cl)c1 C(=O)(C1=C(Cl)CCOC1)N1C(CC(=O)NC2(CCCF)CC2)C2CCC1C2 C(CC(=O)N1CC2CC(O)CC1C2)(C(C)(C)C)NC(CSCCC)=O C1(NC(Cn2cc(C(C)(C)OCC)nn2)=O)NC(=O)N(c2ccccc2Cl)C1=O CC1CN(C(c2sccc2C(F)F)=O)CCC1N=c1[nH]n(C)cc1[N+](=O)[O-] C(CC(C)C)(C(c1nnnn1Cc1ccco1)NCCC1CC1(C)C)OC c1(CC)ccc(Cl)cc1C(N1CCCC1CNC(=O)CNC(=O)COC(C)C)=O N1(C(CCN(CCCCC)C)=O)CC(F)CC1CN(C)C(C1(O)CC(CF)C1)=O c1(C(=O)NC(C(C)NC(C2CCN(CCC)CC2)=O)C)cc(F)c(F)c(C#N)c1 C=C(C)CCCC(=O)NC(CNC(c1c(C)cnn1C)=O)CC(F)(F)F CC1=NOC2(C1)CC(C(N1CCN(C(=O)COc3ccccc3)CC1C)=O)C2 S(=O)(=O)(c1ccc2c(c1)CCCC2)N1CC2N(C(c3cc(C)cc(C)n3)=O)C2C1 c1(C(=O)NC2(C3N(C(C(C)O)=O)CCCC3)CC2)cc2c(cc1Cl)OCO2 N1(C(=O)Nc2ccc(S(N)(=O)=O)s2)CCC2(CCC(=O)N2)CC1 c1(CNC(C2(C)COC(=O)C2)=O)cnn2c1CN(C(=O)C(O)C1CC1)CC2 N1(C(c2cc(C#N)oc2)=O)CCCC(C2CCCN(C(=O)Cc3cccs3)C2)C1 C(=O)(C1CCCc2scnc21)N(C1CN(C(C2CCC(=O)NC2)=O)C1)C C(=O)(CC(C)(C)C(F)F)N1CCN(C(CC(CCC)C)=O)C(=O)C1CC(=O)NC c1(C(=O)OCC(=O)OC)ccc(CNc2cn(CC3CCOC3)nn2)nc1 N1(C(C2(C#N)CCCO2)=O)CC2(COC(CNC(c3ccccc3)=O)C2)C1 c1(C(N2CC(NC(CCCC(C)O)=O)C(C)(C)C2)=O)cc2c(nc1O)CCC2 c1(-c2ccc(CC)nc2)n[nH]c2cccc(C(=O)NCC3COC3)c12 c1(OC)ccc(C(=O)NC2CC(CCNC(=O)C(C)N3CCCC3)C2)o1 c1(CCC)ncc(C(=O)N(CCCOCCNC(=O)C(F)C2CCC2)C)s1 C1(C(=O)NCCCC2(CNC(CCC=CC)=O)CCCC2)CCS(=O)(=O)C(C)C1 Cc1cc(C(=O)NC2C3CCN(C(=O)CCS(C)(=O)=O)C23)cc(C)c1F C1(CNC(CC2(OC)CC2)=O)CCCCN1C(c1ccn(CCF)n1)=O Cc1cc(NCC(C)C(F)F)sc1Br.n12nnnc1CC(C)C2.C(C)C CC1(C)CN(CC2CC(F)(F)C2)CCC1NC(=O)CCCc1nc(C2CC2)no1 N1(Cc2ccc(C)s2)CCOC(CNC(=O)Cc2nonc2C)C1 C1(NC(C(C)(C)OC)=O)CN(c2ncc3cccnc3n2)CC2(CCC2)C1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(CNC(=O)CCCN2CCCC2)C12CCC2 Nc1ccc(C(=O)NC2CC2CNC(c2ccc(Cl)s2)=O)c2ccncc12 c1(C(=O)NC(CC)CN(C(=O)CCC(=O)N(C)C)C)cc(Br)cnc1S c1(OC)ccc(Br)cc1C(=O)NCCN(C(=O)C(n1cc(C)cn1)C)C1CC1 C1(C(=O)NC(c2c[nH]nc2O)C)CCCCCN1C(=O)CC1CCCCN1C N1(C(CCC(=O)N(C)C)=O)CC2(C)CC1C2NC(C1CCSCC1)=O Cc1nc2ccc(C(N3CCC(CCNC(C4COC(C)(C)O4)=O)C3)=O)cn2n1 C1(C)(C(=O)NCC2C(C)CN(C(=O)CCC3CCC(=O)NC3)C2)CCN(C)C1=O C#CCC(C(=O)NCC1=NOCC1)NC(=O)CCC1CCCO1 C1(C(=O)NCC23N(C(c4nnsc4C)=O)CC(CC)(C2)C3)CN2CCCN1CC2 C(C(=O)NCC1CCCCC1NC(=O)CCc1cc(C)on1)(C(C)C)COCC Cc1ccnc(C(=O)NC(C(C)NC(C2CCN(CC3CC3)CC2)=O)C(C)C)c1 n1(C(C)C)ncc(C(=O)NCC2CCN(C(=O)Cc3cc(C4CC4)no3)C2)c1N c1(CNC(C)=O)ccc2c(c1)CCC2NC(c1cnn(C(C)C)n1)=O C12(OC)CCN(C(C3CC4CCC3CC4)=O)C1C2.C1(C(C)OC)CN(C(C)=O)C1 CC1CC(C(=O)NCCOCCNC(=O)CCCOc2ccccc2)CCS1 N1(C(C2C(C)OCCO2)=O)CCN(C(c2cn(CCO)nn2)=O)CCC1C CC1C(NC(c2coc(C(F)F)c2)=O)CCCN1C(=O)C=Cc1cc[nH]n1 CC1(C)CCc2cc(CN3CCOC(c4cccc(C#N)c4)C3)ccc21 C1(NC(C(CC)OCC)=O)CN(C(c2nnc(C)s2)=O)CC1C N1(C(c2cc(OC)ncc2)=O)CC(NC(c2snc(Cl)c2Cl)=O)C(C)(C)C1 C(=O)(C1=CCCC1(C)C)N1CCN(C(c2ccc(C(C)(F)F)cn2)=O)CC1CO Cc1ccc(Cl)cc1C(=O)NC1CCCC(CN(C(=O)Cc2nnc(O)s2)C)C1 C1(NC(c2c(C)nsc2)=O)(CF)CCN(C(C2C(C)(C)C2(F)F)=O)C1 c1(CN2CCN(C(c3scc(CC)n3)=O)CC2C)c[nH]c2cccc(F)c12 Cc1nc(NCCC(C)NC(C2CCCCC2)=O)c2ccsc2n1 c1(C(N2CCCCCC(NC(c3cc(Cl)c[nH]3)=O)C2)=O)cc2cccnn2n1 N1(C(CC#C)=O)CCC(C(=O)Nc2ccc(C3SCCCS3)cc2)CC1 O=S(=O)(c1cc(Br)ccc1Br)N1CCC(N2CCOCC2)C2(CC2)C1 c1(C(N2CC(N(C(C(C(=O)OCC)CC)=O)C)C2)=O)csc2cc(OC)ccc12 CS(=O)c1ccc(C(=O)N(CCNC(=O)C=C2CCSCC2)C2CC2)cc1 CCC(C)C(O)C(=O)NCC1(C(=O)NC(CCO)C(C)C)CC12CCC2 c1(CC(N2CC(CCCCNC(Cc3nc(C)[nH]n3)=O)C2)=O)c(C)nn(C)c1C C(c1ccc(C(F)F)o1)=CC(=O)NCC1CCN(C(=O)CC2(C(F)(F)F)CC2)C1 C1(CC=C)(NC(c2ccc[n+]([O-])c2)=O)CCN(C(=O)C(C)(C)n2cnnn2)C1 c1(C(N(CCNC(CC=C)=O)C2CC2)=O)cc(Br)c(C)s1 CNC1c2ccccc2CCN1C(C1CC2(F)CC1C2)=O C1(CCCNC(=O)COCCNC(=O)CCC2CC2(F)F)CCCO1 c1(SCC(=O)NCC2(O)CCN(C(C(C)CSC(F)F)=O)C2)ccc(F)cc1 C1(NC(CC(CC)C)=O)CCN(C(C2CCCN2C=O)=O)C1(C)C C12(C(N3C(C(=O)NCC4CC(SC)C4)COCC3)=O)CCCN(CC1)C2 N1(C(CC)C(=O)NC(C)CCN(C)C(c2nnsc2C)=O)CCc2ccccc21 C(C(C)(C)CC(=O)N1CCC(CO)C(O)C1)NC(C(C)OCC)=O c1(C(=O)NC(CCCC)(C)C(=O)OC)cc2cc(Br)ccc2c(=O)o1 CC1(C)CCCCC1CC(=O)NCC=CCNC(=O)C(O)Cc1ccc(Cl)cc1 c1(NCCC2CCCN(C(c3nccc(CC)c3)=O)C2)cc(O)nc(=O)n1C N1(C(C2CCN(C(c3cnc(OC)c(C)c3)=O)C2)=O)CCCC2(CCOC2)C1 c1(OC)ccc(S(=O)(=O)NC(Cc2ccc(Cl)cc2)COC)c(Cl)c1 Cc1n[nH]c(C)c1CC(C)C(=O)NCCCN(C(C1CCC(F)CC1)=O)C1CC1 CCCC(CN=c1[nH]c(=NCc2c(CSC)cccc2OC)[nH]c2c1CSC2)OC CCC(C)C(C(=O)N(C)Cc1cc(C)n(C)n1)N(C(=O)C(C)c1cc[nH]n1)C Cc1ccc2[nH]c(C(=O)NCC(C3CC3)NC(C3(N(C)C)CCCC3)=O)cc2c1 c1(C(N(C)CC2CCCN(C(CCSC)=O)C2)=O)c(Cl)cc(C)cc1Cl C(=O)(C(C)(C)c1ccn(C)n1)NCCN(CCOC)C(C1(CO)COC1)=O C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC1CCC2(CN(C(C(C(CC)O)(F)F)=O)C2)O1 N1(C(C2C(NC(C(C=C)(C)C)=O)CC=CC2)=O)CCOCC(C2CC2)C1 N1(CCC)CC(C(=O)N(CCCN(c2nnc(C3CC3)s2)C)C)CC1=O N1(C(=O)COc2cccnc2)CCC2CC2(C(N2CC(O)(C3CCC3)C2)=O)CC1 C1(C(=O)NCCCOC(C)C)C2CCCC2CN1C(c1cccnc1)=O CC#CC1CCN(C(C2CCC(C3CC3)N2C(=O)C=C(C)COC)=O)C1 C1(C(=O)NC2CC(F)(CNC(C(n3cc(C)nc3)(C)C)=O)C2)CCC2(CCC2)C1 N1(C(C2(CCNC(COCC#C)=O)CCC2)=O)CC2CC2(CC)C1 c1(Cn2cc(CC3C(C4CC4)C(=O)O3)nn2)nc2cccc(Cl)c2[nH]1 C1(CC(=O)O)CN(C(=O)CC2CC2)CCN1Cc1cccc(I)c1 C(C1=CCN(C(C2CC(C(F)F)C2)=O)CC1)N.CC(CN1CCOCC1)C(=O)C(N)=O c1(CC)ccccc1NC(C1(F)CC=CC1)=O.C12(O)CC(C1)C(=O)NC2 Cc1cc(Cl)cc(C(N2CC(NC(C3CC(C)(F)C3)=O)CC23CCC3)=O)c1O N1(C(C2CN(CC)C(=O)C2)=O)CCN(C(c2ccnc(CO)c2)=O)C2CCCC12 N1(C(=O)CC2(O)CCOC2)CCCC(F)(C(=O)NC(C23CCC(CO2)C3)C)C1 c1(C(N2CCN(C(C=CC)=O)C(C)C2)=O)cnc2onc(C)c2c1 c1(OC)cccc2c1OCC(C(=O)N(C(C)CN(C)C(c1ccn(C)c1)=O)C)C2 c1(C(N(CCNC(C(c2cccc(F)c2)C)=O)C)=O)ccc(O)c([N+](=O)[O-])c1 C(c1cc(F)c(F)c(F)c1)=CC(N1C2C(NC(C3CC(F)(F)CS3)=O)C(C2)C1)=O c1(C(N2CC(NC(COC(CC)C)=O)(CO)C2)=O)noc2cc(Cl)ccc12 c1(C(=O)NC(C2OCCN(c3ncnc(C)c3F)C2)C)ccc2c(c1)CCOC2 C1(NC(C=C(CCC)C)=O)CCCN(C(C2CCN2CC)=O)C1CC CCCC(CCCNC(=O)C=C(C)c1ccccc1)NC(=O)COC(C)CC CC1CN2CCN2C1.C(=O)CC(=O)NCCC1CCCOC1 c1(OC)cncc(C(=O)NC2CCCCC2CNC(c2cocc2C)=O)c1C CCC(C)(C)C(O)C(=O)N1CCN(C(=O)C(O)CCc2ccccc2)CC1CF N1(C(C2(C)CC(=C)C2)=O)CCCCC(C2CN(C(=O)CCCC(C)C)C2)C1 CCC(F)(F)CC(=O)NC1CN(C(=O)C(CSC)OC)CC1n1ccnn1 C1(C(=O)NCC2(OC)CC(C)C2)CCCCCC1NC(C1CCC(=O)CC1)=O C1(OCCCC)CC(CC2CC2(F)F)C1(C)C.c1(C(=O)O)oc(SC)nc1C c1(C(N2C3C(NC(C4CSC4)=O)CC(C3)C2)=O)cc(F)c(C(F)F)c(F)c1 n1(CC(=O)NCC2(F)CC(CNC(CCC#C)=O)C2)nc(Cl)ccc1=O C(CN(C)N1CCN(CC(C)O)C(C(C)C)C1)c1cnc(C)s1 Cc1nc(CN2CCC(CNC(=O)CN3CCNC(=O)C3)CC2)sc1C N1(C(c2c(OC)cccn2)=O)CC2CCN(C(=O)CCC3(C)CCCOC3)CC12 C1(C(=O)NC(CC)(C)CNC(=O)C(=O)N(C)C)CC2(C1)CC21CCC1 CCC1=NOC(C(N2CCC(C(=O)NCCOC(C)C)(CO)C2)=O)C1 C1(NC(C=CC=CC)=O)CC(NC(=O)CC23CC(C2)C3)C12CCC2 Cn1c(NC(=O)CN2C(=O)CCC2=O)nc2ccc(F)cc12 C1(NC(c2c(OC)scc2)=O)CN(C(c2ccc(F)c(Cl)c2)C)CC1(C)C N1(CC(C2(F)CC=CC2)=O)CCCC2CCCCC12 C1(C(=O)NC(CC)(C)CNC(C2(CO)CCCCC2)=O)CCn2cnnc2C1 c1ccc(C(=O)NCc2cn(CCC)nn2)nc1.C1(C(=O)NC)CCC1OCC Cc1ncccc1-c1cn(CC(N2CCN(C(=O)C3=NOCC3)CC2)=O)nn1.C(C)O C1(NC(C2CCCN2C(c2csc(O)n2)=O)=O)CCC2(CC2)C1 CN1CCC(C)(NC(=O)NC(C2CCCC(O)C2)C2CC2)CC1 C1(NC(=O)NCC(CC(=O)OC)C)C(C)(C)C(NC(=O)OC(C)(C)C)C1(C)C C(=O)(CC(CC)C(C)C)NC1C=CC(CNC(c2c(CC)nco2)=O)C1 C(=O)(C(C)CN(C)C(c1cnns1)=O)NC(CCSCC)C c1(C(=O)NCC(CN(C(c2c(C)nc(CC3CC3)o2)=O)C)O)cnc(Cl)c(N)c1 C(C)(C(=O)NC1CC2CCC1(C(=O)NCCC(N)=O)C2)(C(C)C)NC(C)=O c1(OC)ccc(C(N2CC(NC(=O)OCc3ccccc3)OC(C)C2)=O)nc1Cl N1(C(c2nc(N(C)C)oc2)=O)CC2CC(C(=O)NC34CCCCC3C4)(C2)C1 C1(NC(CC2NCC(C)(C)OC2)=O)N(c2ccnc(C(F)F)n2)CCCC1(C)C C#CCC(CC(F)F)C(=O)NCC1(O)CCN(C(c2cc(C#N)cn2C)=O)CC1 Cc1cc(NC(C2(C)CCCN(C(c3ccn(C)n3)=O)C2)=O)cc(Cl)c1 C1(C(C2(CN3CCOCC3)CCCC2)NC(NOCCC(=O)O)=O)CC2CCC1C2 C1(C(N2CCN(CC(C)(C)NC(C(C=C)C)=O)CC2)=O)CC2(C1)CC(C)C2 C1(O)(C(C)C)CCN(C(c2cn(CCNC(C3(CC(F)F)CC3)=O)nn2)=O)C1 Cc1nc(C)c(C(N2CC(C)(NC(=O)Cc3cccc(C(F)(F)F)c3)C2)=O)o1 C1(CNC2(C(=O)OC)CCC(C)(C)CC2)CCCC2(CCC2)C1 C12(C(N(C3CC(C)C3)C)=O)CCC(CC1)N(C(C1CN3CCC1CC3)=O)C2 c1(CC)c(Cl)nc(C2CCC2)[nH]c1=NCc1ccc2c(c1)COC2 CN1CCCC(O)(CC(=O)NCC2(C)CC(NC(c3cccc(Cl)c3N)=O)C2)C1 C(=O)(C1=C(C)CCCC1(C)C)N1CC2(CCCN(C(CSCC)=O)C2)C1 C1(C(C)NC(COCC=C)=O)CCCN1C(=O)CC(O)C1CCCC1 c1(C(=O)NC23CCN(C(CC=CCC)=O)CC2C3)ccc2ncnn2c1 N1(C(C)=O)CCCCC1C(=O)N(CCCCN(C(=O)C(=C1CCCCC1)F)C)C C1(CC(N2CCC(C)(NC(C3CC(=O)N(CC)C3)=O)C2)=O)(COC)CCOCC1 c1(C(=O)NN2C(CNC(C3CC3CF)=O)CC2)ccc(C(F)(F)F)[nH]1 Cc1cc(F)c(C(N2CCC(CCNC(=O)C(C)n3cnnn3)CC2)=O)cc1F CC1(C)CC(NC(C2CC(=O)CN2C(=O)C=Cc2ccncc2)=O)C12CCC2 c1(C(C)F)ccc(NC(C2(NC(=O)CCCn3ccnc3)CC2(C)C)=O)cc1 c1(C(=O)NC(CNC(C(C)SCC)=O)C(C)C)cnc(C)c(CC(C)C)c1 c1(CNCC(N2CCC(NC(C(CSC)C)=O)CC2)=O)cccc(S(C)(=O)=O)c1 Cc1ccc2cccnc2c1C(=O)NCC1CC(F)(CNC(=O)CC(C)(F)F)C1 N1(CC(c2ccc(OC)cc2)OC)CCN(CCc2ccccn2)C(=O)C1C N1(C(C=C(COC)C)=O)CC2CC1CN(C(=O)CCCCCCSC)C2 CCCCC(CC)CC(=O)N1CCCC1C(C)(C)NC(=O)CC(OCC)OCC C1(NC(=O)C=Cc2ccsc2)CC12CCN(C(c1ccccc1C1CC1)=O)CC2 C=CC(C)(CCOC)C(=O)N1CC(O)CC1CNC(c1cccc(C(C)C)c1)=O N1(C(COCC#C)=O)CCN(C(=O)C(C)N(C)C)C(C)C1 CC(CCCCO)NC(c1sccc1Cl)c1nnnn1C(C)(C)C c1(C(=O)NCCN(C2CCCC2)C(C2CC(CC)C2)=O)ccc2c(n1)CCOC2 C(=O)(C1=C(F)CN(C(=O)C(F)CC2CCOC2)CC1)NCc1onc(C)n1 C1(NC(C(c2cn(CC)nc2)=O)=O)CCCN(C(c2cncn2C)=O)C1C CCCC(CCC)CC(=O)NCCC(C)N(C)C(c1cnn2c1N(C)CC2)=O N1(C(C(=O)NCCC(=O)NC)=O)CCCC(Cc2nccn2C)C1 C1(C(=O)NCc2nc(C)sc2)C2CN(C(c3ccc(-c4cn[nH]c4)cn3)=O)CC12 c1(C(=O)NCC2(O)CCN(C(C(C)(C)CF)=O)CC2)cncc2c1CCNC2=O c1(C(=O)NC(C2CN(C(C3(C)CCCS3)=O)CCO2)C)ccc(N)c([N+](=O)[O-])c1 c1(CC)nnc2c(C(=O)NCC3CC3NC(c3nc(Cl)cs3)=O)cccn12 C1(C(N2CCC(CC)C2)=O)CN(C(=O)C=Cc2cncs2)C2(CCC2)C1 c1(OCCC(N2CCCCC2C2(NC(C3(Cl)CC3)=O)CC2)=O)ccc(F)cc1 C1(C(=O)NCC(C)OCC=C)N(C(=O)CC2CC(C3CC3)C2)CCCC1(C)C c1(C(=O)NC2CN(C(C(CC)C#N)=O)CC23CC3)cnc2c(Br)cccn12 c1(OC(CC)C)cc(N2CC(O)CC2C(=O)NC)nc(C)n1.C12(CC1)C(=O)NC2 c1(C(N(C)CC2(O)CN(C(C(CC)N(CC)CC)=O)C2)=O)cc(F)c(C)cc1F C1(C(=O)NC2(NC(c3nc(C(=O)NCC=C)sc3)=O)CC2)CCC(N(C)C)CC1 C1(OCC(=O)NCC(F)CNC(=O)CCc2cccs2)CCCC1 C#CC1CC2CCC1N(C(C13CC1CN(C(=O)C(C)C(CC)CC)C3)=O)C2 c1(C(N(C(c2ccc(Cl)cc2)C)CC)=O)ccc(N=[N+]=[N-])cn1 C1(NC(C(C)OC(C)(C)C)=O)CCC(CC(=O)NCC2(O)CCN(C)C2)CC1 N1(C(=O)COc2cccc(F)n2)CCCOC(c2ccccc2)C1 C1(C(N(C(CC(=O)N(C(C)C(=O)O)C)C)C)=O)CCN(Cc2ccccc2)CC1 C1(C(=O)NC(CCCNC(c2ncc(C)cc2C)=O)C)CC2COCC(C1)C2 NC(Cc1ccccc1)C(O)C(=O)N1CCOCC1Cc1cccs1 c1(OC)cc(-n2cc(C3(CN(C)C)CN(C(C4CC4(Cl)Cl)=O)C3)nn2)cnc1O Cc1cccc(CC(=O)NCC(=O)N2CC2NC(=O)C(O)CC(N)=O)c1Br c1(C(N(CCN(C(=O)COC2CC2(F)F)CC)CC)=O)cc2c(C)cc(Cl)cc2[nH]1 N1(C(c2c(CC)cno2)=O)CC2CC2(C(=O)N(C2CCC2)CC2CC2)C1 N1(C(C2(C)CCC(=O)NC2)=O)CCC(C2CC2)(CNC(C2CCC(=O)NC2)=O)C1 c1(CC)c(C(N2CC3C(CNC(C4CC4OC)=O)C3C2)=O)nnn1CC c1(C(=O)NC2CC(N(C(CCCCCN(C)C)=O)C)C2)cc(S(N)(=O)=O)c[nH]1 CCCCCCCCS(=O)(=O)N(C1CN(C(c2cccc3[nH]nc(I)c23)=O)C1)C C1([Si](C)(C)C)(CNC(C2(C)CN(C(C3C(OCC)CC3)=O)C2)=O)CC1 N1(C(CN(C2(C)CCS(=O)(=O)C2)C)=O)CC2CC1CN2C(=O)CSC1CC1 Cc1ccc(F)c2oc(C(=O)NC3(CNC(c4cc(F)cnc4O)=O)CC3)cc12 c1(C(N)=O)cccc(OCC(=O)NC2CC(NC(=O)Cc3ccco3)CC2O)c1 c1(C(=O)NC(C)CS)cccc(S(=O)(=O)N(C(C)CC)C)c1.CC(=O)N(C)CCO C1(NC(c2c(C)occ2)=O)C2CC3CN(C(C4C=CCC4)=O)C1C3C2 Cc1cc(C(C)NC(N2CC(C(=O)N(C)C)C2)=O)cc(F)c1 C1(N(C(C(CC)OC)=O)C)CCCCC1NC(c1sc(F)cc1C)=O C(=O)(CC1=CCOCC1)N(C1CCCC1)CCNC(CC(CC)C)=O Cc1cccc2cc(C(=O)NC3CCN(C(c4cc(F)n(C)n4)=O)C34CC4)oc12 c1(NC(C(=O)NC(c2ccc(OC)cc2)CO)=O)ccc2[nH]c(C)c(C)c2c1 Cc1ccc(C=CC(N2CCN(C(=O)CC3CCOC3)CC2C(C)C)=O)cn1 C1(NC(CCCCC=C)=O)CC12CCC(NC(C1CC3C=CC1CCC3)=O)CC2 Cc1ccc(C)c(C(=O)NCC2(C)CCCC2NC(=O)C(C#N)C(C)C)n1 C1(CNC(C(C)OCOC)=O)CCC(F)(CNC(=O)C(O)CSC)CC1 N1(C(C(=O)NCCC)CC(C)CCC=C(C)C)CC2(CCCC2)c2ccccc21 N1(C(CCC2CCC(C)O2)=O)CCC(N)C(F)(F)C1 Cc1cc(=O)c(C(N2CC3CC3(NC(=O)CC3CC=CC3)C2)=O)cn1C n1(CC=C)cc(C(=O)NCCC2CCC(NC(c3cnnn3C)=O)C2)nn1 N1(C(CC(CC)(F)F)=O)CCC2(CCC(NC(c3csc4cncn34)=O)C2)C1 N1(C(C2CCCN(C(c3c(C)ncs3)=O)CC2)=O)CCC2(CCCN2C)CC1 c1(CNC(C(c2nc(CO)co2)N(C)C(c2ccc(Cl)s2)C)=O)cccc(Cl)c1.CO CN1CC2CC(C1)N(C(c1cn(C3(C(=O)O)CCCNC3)nn1)=O)C2 N1(C(c2cnc(C)o2)=O)CCC2(CC1)CC2CNC(C1CCC2CC1C2(C)C)=O N1(C(c2n(C)ncc2)=O)CCC2(CCCN(C(C3CC4(C3)CC43CCC3)=O)C2)C1 c1(C(C(=O)NCC(=C)C)N(C2CC2)Cc2ccsc2)cc(C)c(C)cc1C c1(C(=O)OC)cc(C(=O)OC(C)(C)C)ccn1.N12CCSC(C1)C2=O CCCC(C)(O)C(=O)NCCCCCN(C)C(c1cc(Cl)ccc1Cl)=O C1(C(=O)NCCOCC)(COCC)CCCC1.C(=O)(CCOCC)NCC(N)=O N1(C(=O)CCCC2CC2)CCN(C(=O)CCOc2c(Cl)cccc2Cl)CC(O)C1 N1(C(c2c(CC)n(C)cc2)=O)CC2CCC1C1CN(C(C3CC3C3CC3)=O)CC21 C(=O)(C(F)C(C)(C)O)NCC1(C)C(C)C1 N1(C(C2C=CCN(C(C(C)(C)C(F)F)=O)C2)=O)CC2CCC(CO)(C2)C1 C(=O)(C(Cc1cc[nH]n1)NC(c1cn(C)cn1)=O)N(CCCSC)C C1(CNC(=O)CC2CC(=O)NC2=O)CC2CCC1N(C(C1C3CCCC13)=O)C2 CN1CCOC(C(=O)NC2CC(CCC(=O)NCCc3ccncn3)C2)C1 c1(CN2C(CC)CN(C(=O)CN3CCCCC3)CC2)ccc2c(c1)CCOC2 N#CC1(C2CCCC(C(=O)NC(Cc3cccs3)CO)C2)CCOCC1 C1(CNC(C2(C)CC=CCO2)=O)CC(C(F)(F)F)CCN1C(=O)CCCC(F)F Cc1ccc2cc(C(=O)NC3CCCC(NC(c4ccc[nH]4)=O)C3)c(C)nc2c1 N1(C(CC(=O)NC)=O)CCCC2(CC(NC(c3cc(C(F)F)[nH]n3)=O)C2)C1 CC1CC(NC(=O)CSc2ccc(Cl)cc2)CCN1C(C1CCCC1)=O C(C)(C)(CCC(=O)N1CCCC(N(C(=O)CCSCc2ccccc2)C)C1)OC N1(C(c2ncc(C)nc2)=O)CCCC2C1CCN2C(c1cc(C)n(C)c1C)=O c1(C(C)C(=O)NCC2(NC(C3CC3(C)Br)=O)CCC2)cnn(CCF)c1 CN1CCN(C(=O)CCc2cnn[nH]2)C(CNC(=O)C=C2CCN(C)C2)C1 C1(C(=O)NC(C(C)NC(COCCC(C)C)=O)(C)C)CC(c2ccccc2)=NO1 C1(CNC(Cc2c(C)nc[nH]2)=O)CCCN(C(C2CC(C)CO2)=O)CC1 C1(CNC(=O)CC=C(Cl)Cl)CN(C(C2CC2(F)Cl)=O)CCC12CCC2 C1(CC(C)C)CN(C(=O)CN(C)S(=O)(=O)N(C)C)CCN1C(=O)C(O)C(F)F C1(CNC(CCC)=O)CCN(C(=O)CC2CCOC2C)CC1 C(=O)(C(CCC(C)C)NC(C1CC(C)(C)CCO1)=O)N1CC(C)C=C(C)C1 C1(COC)COCCN1C(=O)C(C)(C)CNC(=O)Cc1ccn(C)c1 Cc1ncc(CCC(=O)NC2CCC(CNC(c3ccc[nH]3)=O)CC2)c(O)n1 Cc1cc(C(=O)NC2CCC(Cn3cc(C4OCCO4)nn3)CC2)c(C)s1 CCCCC(CNC(C1CCCCN1CC(F)F)=O)NC(c1[nH]c(C)nc1C)=O CN(CCCC(=O)NC1CCCCCCC1NC(=O)C(C1CCCCC1)F)N=O N1(C(C(C)SCCCC)=O)Cc2n[nH]cc2C1C(=O)NCc1cc(C(C)C)n[nH]1 N1(C(c2ccc(C)c(Cl)c2)=O)CC(C)CN(C(=O)Cc2cc[nH]c(=N)c2)CC1C N1(C(CCOCCN(C)C)=O)CCC2CCN(c3nc4ccccc4o3)CC2C1 C1(c2nnnn2CCCF)(N(CCC2C(=O)NC(=O)N2)C2CC2)CCC2COC1O2 C1(C(C(=O)NCC2CC2(F)F)C2(C(=O)OC)CC2)CC2(CCC2)C1.C(=O)(COC)N c1(C(=O)NCC(C)CNC(c2cnn[nH]2)=O)scnc1Br C(=O)(C1=CS(=O)CCC1)NC(C)CN(C)C(c1ncoc1C1CCCO1)=O CCC(CC)C(C)C(=O)N1CC(CNC(=O)CC2CNC(=O)O2)C(O)C1 c1(-c2scc(NC(Cc3nc(COC)sc3)=O)n2)cccc(F)c1F N1(C(c2c(CC)cc[nH]2)=O)CC2(C1)CN(C(C13CCC(C1)C3)=O)CCO2 O=C(NNc1ccccc1C(F)(F)F)Nc1ncc2ccc(Br)cc2n1 N1(CC(N2CC(SC)C2)=O)CCN(C(c2cncc(C)n2)=O)CC1=O N1(C(c2n[nH]c(C)c2Cl)=O)CCC(NC(c2ccc[n+]([O-])c2)=O)C12CC2 C1(NC(c2c(COC)cco2)=O)CC2(C1)CN(C(=O)CCC1CC1(C)C)C2 c1(C(N2CC(CCC)N(C(=O)C(C)N(C)C)CC2)=O)cc2c(nn1)OCCS2 c1(-n2c(CCC)nc(-c3ccc(NC)cn3)n2)ccc(Br)c(C)c1 N1(C(C2CCN(C)CC2)=O)CCOC2CN(C(=O)CN3CC4CC4C3)CC12 C1(C(=O)NC(C2(O)CN(C(=O)C3=COCC3)C2)C)CCc2cn(C)nc2C1 N1(c2nc(C)nc(-c3ccco3)c2)CC2CC1CN(C(C1CC1F)=O)C2 C1(C(N(CC)Cc2cncn2C)=O)CC(NC(c2csnc2Cl)=O)C(O)C1 N1(C(c2ccc(SC)o2)=O)CCOCC1C(=O)NC(C(N)=O)C1CCCC1 CC1Oc2c(C(=O)NCCCC(C)NC(=O)C(C)(C)CF)cccc2NC1=O c1(CC(N2CCN(C(C(C)=C3CCCC3)=O)C3C2C3)=O)cc2ccccc2o1 C(C)(C)(CC(F)C(=O)NCCc1nc(C)no1)NC(CC(CC)C1CCC1)=O N1(C(CC2CCC(C)(C)CO2)=O)CCN(C(c2ccns2)=O)C2CCCC12 N1(C(CC(=O)NCC2CC2)=O)CCC(C(C2CC2)NC(=O)CC2CCC2)CC1 N1(C(c2ccc(F)c(Br)c2)C(=O)NCC)C(C)CCC(C(=O)OC)C1C c1(C(C(=O)NCC2C(CNC(=O)CCF)C2)O)ccc(Cl)cc1Cl S(=O)(=O)(CCC(=O)N1CCC(C(C)NC(c2cncc(N)c2C)=O)C1)NC c1(C(=O)NC(CC=C)CNC(=O)CN(CC)CC)ccc(F)c2ncccc12 N1(C(c2ccc(Cl)cc2)=O)CCC(NC(c2c(C(C)C)nco2)=O)C(C)C1 c1(CC)nc(C(=O)NCC2CCC(NC(C3CN(C)C3)=O)C2)cs1 C1(C(N2C(CCNC(c3n(C)ncc3Cl)=O)CCCC2)=O)CCCC2(CCC2)O1 c1(NC(CC=C)CNC(=O)CC(C)(C)CCOC)ccnc(S(C)(=O)=O)n1 CCCCCC(CC)C(=O)N1CC(CNC(C2CCOCC2(C)C)=O)C(C)C1 CC1CCC(C(=O)NCc2ncccn2)N(C(=O)CCc2cnn(C)c2)C1 c1(C(=O)NC2C(OC)CN(C(c3c(Cl)n[nH]c3C)=O)C2)nccc(N)c1Cl C1(C(NOC(c2ccncc2)C)=O)C=CCN1C(C1CC1F)=O C1(NC(c2c(C)nns2)=O)CCCCC1NC(c1ccccc1F)=O C1(CCNC(=O)C(=C2CCCCC2)F)CCCN1C(=O)Cn1ccc(C(F)F)n1 C(=O)(C(C)CC(C)(C)C)N1C(SCC)C(NC(c2cc(C)nnc2O)=O)CCC1 C1(CNC(=O)C(c2ccccc2)F)(CO)CCCN(C(C2CC2[N+](=O)[O-])=O)C1 c1(NC(C23CC(CNC(CCCC#C)=O)(C2)C3)=O)cc(C)ccc1CC CC(C)CC(CNC(C1(c2ccccc2F)CCC1)=O)NC(=O)CS(N)(=O)=O c1(CC(C(=O)NC(C)CCc2ccccc2F)N)cccnc1F N1(C(C(C)C#N)=O)CCC2(CNC(c3scnc3C(C)(C)C)=O)CCCCC12 CC1CC(NC(c2ccc(CO)o2)=O)CN1C(c1sc(F)cc1Br)=O c1(C(=O)NCC(c2cnn(C)c2)NC(C(C)C2CC2)=O)ccc(C(O)CF)cc1 C=CCC(C(=O)N(C1CCCCN(C(=O)COCP(C)(C)=O)C1)C)C(C)C C(=O)(C1CCc2cccc(O)c21)N1CCC(CCNC(CC(C)N(C)C)=O)CC1 N1(C(C2(SCC)CC2)=O)CC(CO)C2(C1)CN(C(C1CC3(CC3)CO1)=O)C2 c1(NC(C(=O)NCc2cc(C)cc(C)c2)=O)cc(Br)cc(F)c1F N1(C(CC=CC(C)(C)C)=O)CCC(CCNC(=O)CS(C)(=O)=O)C(F)(F)CC1 C1(C(=O)NCC2(F)CC(CNC(C)=O)C2)CCCC(C)(C)CC1 c12cc(ccc1NCC1(OC)CC(C)C1)C(c1nnnn1C)N2.C(C)(=O)OC N1(C(Cn2c(C)cnc2)=O)CCCC(CNC(=O)C(C)C(F)F)C1 c1(C(N2CC(C(C)NC(C3C(C=C(C)C)C3(C)C)=O)C2)=O)cc(C)ncc1C c1(C(=O)Nc2ccc(NC(=O)C3CC3)c(O)c2)c[nH]c2ccc([N+](=O)[O-])cc12 CC1(C)OC2CC(C(N3CCCCC3CNC(=O)CC3(O)CCCC3)=O)CC2O1 CCC(C)(CC)C(=O)N1CCC(NC(C2CCC(F)(F)CC2)=O)C(O)C1 c1(C(N2CC(OCCN(C(COCCN(C)C)=O)C)C2)=O)cc(C2CC2)[nH]n1 C1(C)(CC(=O)NCCC2(OC)CCC2)CCN(C(c2cc(C)co2)=O)C1 c1(N2CC(O)(CN(C(C(C)C3CCCO3)=O)C)C2)ncc(Cl)cn1 c1(C(=O)NCCOCCN(C(C(c2ccccc2)C)=O)C)c(O)cc(O)cc1O c1(OC)ccc(C(N2CCC(N(C(=O)CN(C3CC3)CC)C)C2)=O)c(C)n1 Cc1cc(F)c(C(N2CCC(F)C(NC(=O)C(=O)NCC3CC3)C2)=O)cc1F c1(CC)cc(CC(N2CC3CC3(CNC(C3COCCN3C)=O)C2)=O)n(C)n1 C1(C(=O)NC(CNC(CCOCC(C)C)=O)C2CCC2)COCC(C)(C)O1 C(CCCCCF)NC(C1CC2CC1(c1ccc(F)cc1)C2)=O c1(OC)c(C(=O)NC(CNC(c2ccncc2O)=O)CC(C)C)sc(Cl)c1Cl N1(C(C2(C)CC3(CC3)C2)=O)CC2CCC1CC2NC(=O)C(c1ccccc1)F C1(NC(CCCC#C)=O)C(C)CCN(C(c2ccc(-c3ccco3)o2)=O)C1C N1(CC(=O)NC2C(CCC)CN(C(C3CCCCN3C)=O)C2)CCCNS1(=O)=O N1(C(=O)NCCCCCN(C)C)CCC(O)(CO)CC1.C1(C(C)C)CCCC1C(=O)N c1(OC)ccc(C(N2CC(NC(=O)C3=CCSC3)C(C)C2)=O)n2nccc12 Cc1cc(CC(N2CC(CNC(c3[nH]c(O)nc3C)=O)CC2C)=O)cc(C)c1 C1(CCNC(=O)CCC2CCC2)CCCN(C(C2CCC(C(N)=O)O2)=O)C1 C12CCCN1C2=O.c1(CNC(C(C)NC(C2CN(C(N)=O)C2)=O)=O)ccccc1 Cc1ccc(-n2cc(C(=O)NCC(CO)NC(c3ccc(O)cn3)=O)nn2)cc1 C(=O)(CC(CC)CCCC)N1CCCC(CC(N2C(CCC=C)CCC2)=O)C1 c1(CC(C)C(=O)N2CC(NC(c3ccccc3OCCF)=O)C2)cccc(F)c1 n1(CC(=O)NC2CCC(NC(c3nnn(C)n3)=O)CC2)nc2n(c1=O)CCSC2 c1(C(N2CCCC(C(C)NC(C3CCOC3)=O)C2)=O)ccc2c(c1)OC(C)(C)O2 c1(CCC(=O)NC(CNC(CC(C)c2cnn(C)c2)=O)C)ccc(Br)cc1 N1(C(C2(C(N(C)C)=O)CC2)=O)CC2CC2(CNC(c2c[nH]nc2F)=O)C1 c1(C(=O)NCC(C)CN(C)C(C2COC(=O)N2)=O)ccc(OCC(F)F)cn1 N1(C(C2CC(NC(c3c(F)ccc(C)n3)=O)C23CCC3)=O)CC(C2CCCC2)C1 N1(C(C2ON=C(CC)C2)=O)CCC2(CCCN(C(=O)CC3CCC(C)C3)C2)C1 C1(CC(=O)N(C(C)CCNC(=O)C(C2CCOCC2)F)C)CCCCN1C n1(CCC)nnnc1C(c1ccc(C(=O)OC)o1)NCC.C(=O)OC CC1=C(C(=O)N2CCC(N(C)C(c3cc(N)c(O)c(F)c3)=O)C2)CCC(C)(C)C1 c1(CC(=O)NCC2(C(N)=O)CN(C(c3scc(C)c3)=O)C2)cc2ccccc2o1 C(=O)(C(C)(C)CC(=O)NC1CC=C(C(=O)N(C)CCC2CCOCC2)C1)OC c1(C(C)NC(=O)OC(C)(C)C)nc(C)c(C(=O)N(C(C)C)CC)s1 Cc1cc(N2CCCCC2)ccc1NC(=O)CC1CCC12CCC2 N1(C(C2(NC(=O)COc3ccccc3)C(C)(C)C2)=O)CC2(CCC2)C1 C(=O)(CCC(CC)NC(C1(C)CCCCCC1)=O)N(CC#C)Cc1ccco1 c1(C(N2CC(CNC(C(C(COC)C)C)=O)C2)=O)c(Br)ccc2n[nH]cc12 Cc1cc(=NC2CN(C(c3cccn(O)c3=O)=O)CC2C)[nH]c(Cl)n1 N1(C(CCc2ccc(=N)[nH]c2)=O)CCN(C(=O)C2=CCCCC2)C2CC12 c1(C(=O)NCCN(C(C2C(SC)CCC2)=O)C)cnc2c(ccn2C)c1 c1(C(N2CC(NC(C3(CC#C)CCC3)=O)C(C)C2)=O)cc2ccc(Cl)c(F)c2[nH]1 N1(C(COCC(C)(C)C)=O)CCC(C2CCN(C(c3cccnn3)=O)CC2)CC1 C1(C(=O)OC(C(N(OC)C)=O)C)CC2(CCCCC2)C1 C(=O)(CCS(=O)(=O)N(C)C)N(C1CCC(NC(=O)CC2CCNC2=O)CC1)C CC1CCCC1(C)C(=O)N(C)CC=CC(=O)NCc1nc(=O)o[nH]1 N1(C(c2ccc(CCCCC)s2)=O)CCC(C)(CNC(C2C(C)C2C)=O)C1 c1(CC(=O)NC2CCN(C(CCCSC)=O)CC2C(C)C)c(C)cc(C)cc1C c1(C2CCN(C(c3ncsc3C(F)(F)F)=O)CC2)ccc(F)c(F)c1 C1(C(=O)OCCC=C=C)CCc2nc(C)ncc2C1 C1(C(=O)NC2(C)CC(F)(F)C2)CC(NC(c2cnns2)=O)C12CCC2 C1(OC)CCCCC1CNC(=O)CC(C)(C)NC(c1nc(C)oc1C)=O Cc1ccc(F)cc1CC(=O)NC(CN(C(=O)CN1CC2CC2C1)CC)C1CCC1 Cc1cccn2cc(CC(=O)NCCNC(C3(CF)CC3)=O)nc12 c1(C(=O)NCC(C(N2CCC(C=C)C2)=O)OC)ccn2nccc2c1 C1(C2C(=O)N2)CCN(CC)CC1.C12(NC(c3ccncc3)=O)COC(CSC)(C1)C2 c1(C(=O)NC2CN(C(=O)CCc3cncnc3)C2)ccc(C(F)(F)F)cc1 c1(C(=O)NC2C(CC)CN(C(=O)C=CC(=O)NC3CC3)C2)cc2ccccc2[nH]1 C1(C(=O)NC2CCCN(C)C2)(NC(c2cc(C#N)cn2C)=O)CCC(C)(C)C1 c1(CC(N2CC(C)C(NC(=O)C(F)(F)c3nccn3C)C2)=O)cccc(O)c1F N1(C(C2(NC(N)=O)CC2)=O)CC(NC(c2c(C)sc(O)n2)=O)CC12CCOCC2 C=CC(C)CC(=O)NCC1(C)CCCN1C(c1csc(-c2ncccn2)n1)=O C(=O)(C1CCCc2cncn21)NC1C(NC(c2ccn(C)c2)=O)COCC1 CC(C)C(F)C(=O)NC(CC1CC1)C(N1CCOCC1CC1CC1)=O N1(C(=O)Cc2cccc([N+](=O)[O-])c2)CCC2C1CCCN2C(C1CC(O)C1)=O c1(OC(C)C)ccc(N)c(C(=O)NCC2CN(C(c3csc(C#N)c3)=O)C2)c1 Cn1cc(C(=O)NCCc2ccc(C(F)(F)F)nc2)c2cccnc12 C1(NC(C(n2c(C)cc(C)n2)C)=O)CCN(C(c2ccc(N)cc2F)=O)C(C)C1 C(C)(CCCC(=O)N(C)CC1(C#N)CCC1)NC(C1C(CCC)C1)=O C1(N(C(=O)CC2CC3(CC3)C2)C)CCC(NC(C2CC2C2CCCO2)=O)CC1 c1(C(N2C(C)(C(=O)NCc3c(C)n[nH]c3)CCC2)=O)c[nH]c2ccccc12 CC(C)(C(F)(F)F)OCC(=O)N(CCNC(=O)CCC1CCC(=O)N1)C1CC1 c1(C(=O)NC(C(C(C)C)NC(c2cc(C3CC3)[nH]n2)=O)C)ncc(Cl)cc1Cl c1(NC(C2N(C(c3ccc(OC)cn3)=O)CCCC2)=O)cc(OC)ncc1F CCC(C)C(C)C(=O)NCCC(C(C)C)NC(=O)COC C(=O)(C(C)C(=O)OC(C)(C)C)NC(C(C)C)CNC(=O)C(Cl)=CCl C1(NC(C2C3CCOCC23)=O)CN(C(c2c(F)cccc2Br)=O)CCC1F c1(C(N2CC3C(C(=O)Nc4nc5c(s4)CCC5)C3C2)=O)ccc2cccnn12 C1(NC(C2C(CC)CCC2)=O)CC(C2CCN(C(=O)CCCF)CC2)C1 c1(C(=O)NC(CC)CNC(=O)CCc2ccncn2)ccc(OC(F)F)nc1Cl C(=O)(C1=CCCCC1)NC=O.N1(C(C)=O)CCCC1C1CC1.CC1C=CC1 C1(C(N2CCC3(CSC3)C2)=O)CC(c2nc(OC(C)C)no2)CCC1N c1(C(=O)NC2CCN(C(CC(CC)C3CC3)=O)C2)[nH]c(C)c(S(N)(=O)=O)c1C N1(C(Cc2cncc(C)c2)=O)CCN(C)C(CNC(c2cnc(C(N)=O)s2)=O)C1 CCC(C)(CNC(c1ccccc1)=O)C(=O)N1CCC(O)CC1CO C12(C(=O)NCCC3CCN(C(c4nc(C)sc4)=O)C3)CC1COC21CCC1 C1(C(=O)NC(c2ccncc2F)C)CC(O)CCN1C(c1cnn[nH]1)=O N1(C(c2ccc(C(=O)OCC)cc2)C(=O)NCCC)CC(OCC)CCC1C C1(O)(c2cn(C(CNC(c3c(C)[nH]c(=N)s3)=O)N(C)C)nn2)CC2CCC1C2 n1(CCCC)ccc(C(=O)NC(C)CCN(C(=O)Cc2ccoc2C)C)n1 c1(C(N(C)CC2CCN(C(CNC)C)CC2)=O)cc2cccc(OC)c2o1 c1(CNC(c2ccc(OC)o2)=O)cccc(C(C)C)c1.C1(SC)CC1CNC(=O)CO N1(C(c2c(CCNC(c3nn(C)c(Cl)c3)=O)n[nH]c2)=O)CC(=O)N2CCCC2C1 c1(C(=O)NC(CNC(C2C(C(=O)OCC)C2)=O)C)cnccc1-n1cccn1 C1(CC)CC(C(=O)OCC2CCCCC2(F)F)CCC1=O N1(C(C(C)OCC)=O)CC(C)(C)CC1CNC(c1ccc(CC(F)(F)F)cc1)=O CC(CCCNC(=O)C(C)(C)N1CCC1)NC(c1cn(-c2ccccc2)nn1)=O C1(C(N2CCC(OCC(C)C)C2)=O)(CNC(C2CC(F)(F)C2)=O)CC12CCC2 CC1(OCC(=O)NCC2(NC(C3(O)CCOC3)=O)CCC2)CCOCC1 CC(C)C(C(=O)NC(C)(CNC(=O)CCc1ccsc1)C1CC1)N1CCCC1=O C1(C(=O)NC2C(NC(CNC(=O)CC(F)(F)F)=O)CC2)CCc2ccnn2C1 CCN=c1[nH]c(C(N2CCC(CNC(c3cnn(CC(C)C)c3)=O)CC2)=O)cs1 C1(CC)CCN(C(=O)CC2CCCC(C)C2)C1CNC(c1sccc1C)=O C(=O)(N1CC=CCO1)C1(CO)N(Cc2c(C(C)C)noc2)CCC1 N1(C(C2(OCC)CCCC2)=O)CCN(C(c2cccn2C(C)C)=O)CC1C1CC1 Cc1nc(C)c(C(N2CCC(C)(NC(c3ccc(C(F)(F)F)[nH]3)=O)C2)=O)o1 c1(CC)ccc(NC(=O)C(O)C2CN(C(=O)CCC3(C#N)CCC3)C2)cc1O C1(C(N2CC(C)N(C(c3nnsc3N)=O)CC2)=O)CCc2ncccc2C1 C=C(C)C(C)(C)C(=O)NC(CN(C(=O)CSc1ccccn1)CC)CC C1(CNC(CCC#CC)=O)CC2CCC(C1)N2C(=O)CC1CC2(CCCC2)CO1 C1(C(N2CCC(n3cnnn3)C2)=O)CSCN1C(c1cc(C(F)F)no1)=O CCC(CNC(=O)C(CC(C)C)NC(=O)C(C)N(CC)CC)CC(C)C CC1(C)CC(NC(=O)Cc2ccc(C#N)cc2)CN1C(C1C2C3CCC(C3)C12)=O c1(C(N2CC(F)(CNC(CS(CC)(=O)=O)=O)C2)=O)nn(C)c2ccc(F)cc12 C#Cc1cc(F)c(C(=O)NCCc2ocnc2CNC(=O)CCOC)c(F)c1 c1(C(=O)OCc2cnc(=N)[nH]c2)ccc2ocnc2c1 Cc1ncc(C(N2CC(F)(C(=O)NCC(CO)C(C)C)C2)=O)c(=N)[nH]1 C1(C)(C(N(CC(C)(C)NC(C(c2cnn(C)c2)C)=O)C)=O)CC=CCO1 C1(NC(C2(CC#C)CC2)=O)CC(CNC(c2occc2C)=O)C1(C)C N1(C(C(CCC)C)=O)CCN(C(=O)CSc2ccc(Cl)cc2)CC1c1cn[nH]c1 C(=O)(CC(C)c1cnn(C)c1)NCCN(CCOC)C(C1CC1(C)C)=O Cc1nc(C)c(CC(=O)NC2(CF)CCN(C(=O)C(C)c3ccsn3)C2)c(O)n1 Cc1cc(C)c(C(=O)N(CCNC(C2(c3ccno3)CC2)=O)CC2CC2)c(O)c1 c1(C(=O)NC2CCN(C(CCC(N)=O)=O)CC2F)ccc2nc[nH]c2n1 CC1(C)OC2(CO)CC1(C(N1CCC(NC(C3(Cl)CC3(F)F)=O)CC1)=O)C2 CC1CN(C(c2cnc(O)s2)=O)CC1NC(=O)CCCNC(c1ccc(F)cc1)=O C(=O)(CC1CCc2ccccc21)N1C2C(CNC(=O)CC3CSCCO3)C(C2)C1 c1(-c2nc(CC(CCOC)(C)C)on2)cccc(Cl)c1OC C1(C(N2CC(C)(C)CC2C)=O)CN(C(=O)C=CCN2CCCC2)CCC1(C)C c1(OCCNC(=O)NC2C(c3ccn(C)c3)C2)cc(F)ccc1F c1(SCC(C(=O)N(C(C)C)CCNC(=O)C(C)(O)C2CCC2)C)ccc(F)cc1 Cc1cc(NC(=O)C(C2CCCN(C(C3CCCCO3)=O)C2)(C)C)c(C)s1 S(=O)(=O)(c1cnccc1NCC(c1cccs1)C)N1C(COC)C=CC1 N1(C(C(C2CC=CCC2)NC(C=CCOC)=O)=O)CC2C3C=CC(C3)C2C1 c1(C(=O)Nc2coc(-c3ncccc3Cl)n2)cccc(Cl)c1F c1(C(C2CCCC2)C)cn(CCCSCCN)nn1.C(=O)(CSC(F)F)N(C)CCC1CC1 c1(C(=O)NCC2CCN(Cc3ccc(COC)o3)C2)noc2c1COCC2 Cc1ccc(CCC(C2CC3C=CC2C3)=O)c(F)c1.C123CC(C1)(C2)NC3=O c1(C(=O)NCC(CC)(C)NC(C2CC3CCC2CC3)=O)ccc2ncccc2n1 N1(CC)CC(NC(C2CC(=O)CN2C(C2(O)CCOC2)=O)=O)C(C)C1 CCCC(CC(C)C)C(=O)N1CCC2(CC1)CC2NC(C1CCC1)=O C(=O)(C(F)C(=O)NCC1CC(OC)CN1C(c1csc(Cl)n1)=O)OCC N1(C(C=CCOCCOC)=O)CC(NC(c2cc(Cl)c(Cl)s2)=O)C2CC2C1 C#Cc1cncc(C(=O)NC(C2CCCN2C(c2csnc2C)=O)C)c1 c1(C(=O)NCC2(N(C(=O)CC3CC3)C)CC2)ccoc1C1CC1 Cc1cc(Cl)ccc1NCn1c(C2(Cc3ccco3)CCC(=O)N2C)nnn1 Cc1nc(N2C3CCC2C(CNC(c2ccc4cc[nH]c4n2)=O)C3)ccc1C#N C(=O)(C(C)CC(F)F)NCC(C1CCCN(C(CCc2ccc(C)o2)=O)C1)C c1(C(=O)OC)cc(NCC(C)N(C(=O)C(CC)n2ccnc2)C)ncn1 c1(C(=O)NC2C(NC(Cc3ccc(CC)cc3)=O)COCC2)nnc(O)nc1O c1(CNC(N2CCC(N(CCCCOC)C)CC2)=O)cccn(C)c1=O C(=O)(C1=NOC2(CCC2)C1)NCC1C=NCC1.C12CC3CCC(C1)N3C(=O)CN2 C1(O)(C(=O)Nc2ccc(N3CCCN(CC)CC3)nc2)CC12CCOCC2 CCC(C)CCCCC(=O)NC1(C2CN(C(=O)C(CCSC)OC)C2)CC1 c1(CNC(CN(C)C)=O)ccc2c(c1)CN(C(=O)C=CC=C(Cl)Cl)C2 C(C)(CC(C)C(F)F)NC(C(C1CN(C(c2ccnc(C)c2C)=O)C1)OC)=O CC1CN(C(=O)C(F)(F)F)CC1(C)C(=O)NCCCNC(c1ccsn1)=O n1(C(CC)(C)C)nnnc1C(CSC1CC1)NCc1ccco1.c1(C)cccs1 C1(CCC)CN(C(c2cn(C)nn2)=O)CCN1C(=O)Cn1cnnc1 N1(C(c2nc(-c3cn(C)nc3)oc2)=O)CC2CCC(C1)N2C(=O)CC1(C#N)CC1 Cc1cc(C(N2CC3CC2CC3CNC(=O)C=CC(C)C)=O)c2ncccc2c1 C1(NC(C2(NC(C3CCN(CC)CC3)=O)CC=CC2)=O)COCC(C)(C)C1 CCCCC(CNC(=O)CNC=O)NC(=O)Cc1cnccn1 C1(CNC(c2ccc(Cl)cc2)=O)CC2(CCN(C(=O)C=CC3CC3)CC2)CO1 CCCC(C(=O)NC1CCN(C(C2(COCC)CCCC2)=O)CC1F)C(C)C c1(C(N(C(CNC(c2cc(CC)on2)=O)C)CC)=O)ccc(C)c2ncccc12 N1(C(C2N(C(C)=O)CCCC2)=O)CC(N=c2cc(C)[nH]cc2C#N)C(C)(C)C1 C1(NC(N2CCC(C(F)(F)F)C(F)(F)C2)=O)C2Cc3ccc(Br)cc3C12 CC12CSCC1CN(C(C1CCN(C(c3cc4cccnc4s3)=O)O1)=O)C2 c1(C(N(C(C)CNC(=O)CNC(c2cscn2)=O)C)=O)cn(C)c(=O)n1C c1(NC(=O)NC(c2ccccc2)CCOC)ccc(C)c2c1CCC2 CC1(C(=O)NCC2(CNC(C3CCCCC3F)=O)CC2)COc2ccccc2O1 c1(C(=O)NCCN(C(COCC#C)=O)CC)ccc(N)c([N+](=O)[O-])c1 c1(C(N2CC3CCN(C(C4CC4F)=O)C3C2)=O)cc(Br)c2ccccc2n1 CC1CN(C(C23CC(O)C2C3)=O)CCC1NC(c1nnc(S)n1C)=O C(=O)(C(CC=C(Cl)Cl)c1ccccc1)N1CCC(NC(c2cnsn2)=O)C12CC2 C1(NC(C2CCS(=O)(=O)CC2)=O)(CO)CCCN(C(=O)C(c2ccccn2)O)C1 CC1CN(C(c2[nH]nnc2C2CC2)=O)CC1(C)CNC(c1ccc(F)c(F)c1)=O c1(C(C)C)ccc2cc(C(=O)NC(C3CCCC3O)C)[nH]c2c1 n1(CC)nc(C)c(CC(=O)NCC2(F)CN(C(=O)CC(C)(O)COC)C2)c1C N1(C(C2(CC)CC2)=O)C2CCC1CN(C(c1ncoc1-c1cnn(C)c1)=O)CC2 C1(C(C)NC(=O)CCCN2CCCCC2)CCCCN1C(C1CCCC1C)=O Cc1sc(NC(C2(C)CC(c3ccccc3)C2)=O)nc1C(=O)O C1(NC(COCCCC)=O)CCC(C(=O)N(CCCCO)C)C1 C1(C(N2CC(C=C)C(NC(=O)Cc3cn[nH]c3)C2)=O)CC(c2ccccn2)=NO1 c1(COC)nc(C(=O)N(C)CCOCCNC(=O)CCCc2cccs2)n[nH]1 C(=O)(CCCCCNC(C1CCCCS1)=O)N1CCC(OCC)C1 C(=O)(CC(C)C(C)C)NC1(COC)CN(C(=O)Cn2ccnc2C)C1 C(=O)(C(C)C(F)(F)C(F)F)N1CC(SC)C(NC(=O)CCn2ccnn2)C1 N1(CC(N2CCC(N(C(=O)Cn3ccsc3=N)CC)C2)=O)CCCCC1C C1(C(N2CCC(CNC(c3coc4c3CSC4)=O)C2)=O)CCCCC12OCCO2 C1(NC(C(C)c2cccs2)=O)CC12CC(NC(=O)COC1CCCC1)C2 CC(C)CC(C)CC(=O)N1CC2(NC(=O)CCC(C)(C)C)CCC1CC2 C1(C(N2CC3C(CNC(=O)COCC(F)F)(C3)C2)=O)CC12CCCCCC2 N1(C(=O)OC(C)(C)C)CCC(COC(c2ccc3ncsc3c2)=O)CC1(C)C C1(NC(C(C)Br)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)c(F)c1)C N1(C(COCCCC)=O)CCOCC1CNC(C1CC(CN(C)C)C1)=O c1(OC)ccc(C)c2[nH]c(C(=O)NCCC3CN(C(=O)C(C)C)C3)cc12 C1(F)(COC)CC(NC(=O)C(=O)NCC(c2ccccc2)C)C1 N1(C(c2cncc(C)n2)=O)CCC2(CCN(C(=O)C(C3CCCCC3)F)CC2)C1 c1(C(C)=O)cccc(OCC(=O)NCCCCCN(C)C(C2(SC)CC2)=O)c1.C(F)F C1(F)(CNC(Cc2nc(C)sc2)=O)CCN(C(=O)CS(C)(=O)=O)C1 c1(OCC)cc(C(=O)N(C2CN(C(c3ccc(CC)cc3)=O)C2)C)cc(Cl)c1O C1(NC(CC(COC)C)=O)CN(C(=O)CCCC2CCCO2)Cc2nccn2C1 C1(F)(C(N2CC(C(C)NC(CSC)=O)OCC2)=O)CC2(CCC2)C1.C(COC)O c1(C(=O)NC2CCN(C(C3CC4CCCCC34)=O)C2)ccn2cnnc2c1 c1(N2CC(COC)N(C(c3ccsc3)=O)CC2)ncc2c(Br)cccc2n1 N1(C(c2c(Br)cn(C)n2)=O)CCC2(NC(c3ncccc3Cl)=O)CC2C1 c1(CNC(CCNC(=O)OC(C)(C)C)=O)cccc(C(C)(C)CO)c1 C1(O)(C(=O)OC)CCN(C2CCN(c3ccc(Cl)cc3)C2=O)C1 C1(CCNC(C(CC)=CC)=O)CCCN(C(c2cn(CC)cn2)=O)CC1 C(=O)(C1CCCc2scnc21)NCC1CCN(C(C(CC)n2ccnc2)=O)CC1 Cn1cnc2cccc(C(N3CCOC(Cc4ccccc4Cl)C3)=O)c12 N1(C(C(CC)N(CC)CCOC)=O)CC(O)CC1C(=O)NOCC=CCl CCC(CC)(C(=O)NC1CN(C(C2CCCCC2N=[N+]=[N-])=O)CC2CC12)C(C)C c1(NC(COCC)=O)ccc(NC(c2cccc(OC(F)F)n2)=O)cc1C#N c1(NC(C(c2c(C)n[nH]c2C)C)=O)ccc2c(c1)C(=O)NC2=O c1(C(C2CC2)NC(=O)Nc2nc(-c3ccncc3)cs2)c(C(F)(F)F)cccc1Cl C12(NC(c3cn(CC)nc3)=O)CCC(CC)(C1)OC2.C1(C(=O)N)CC2CC(=O)C1C2 C1(OC)CC(C(N2CC(O)(CCNC(=O)C=CC3CCCC3)C2)=O)C1(C)C CCC(C)CC(C(=O)NCCC1(C)CCOC1)NC(c1cccc(=O)o1)=O N1(C(c2c(C)cc(O)cc2C)=O)Cc2ccc(C(=O)NC3COC(=O)C3)cc2C1 O(N(C)C(=O)C(C)(CNC(c1cc(C)c(CC)o1)=O)CC)CC(=O)OC c1(SCCC(=O)N(CCNC(c2cc3cscc3s2)=O)CC)ncnc2[nH]cnc12 c1(OC)cc(CN2CC3CC2CN3C(c2[nH]cc3c2CCC3)=O)cc(F)c1O C1(CC(=O)N(C(C2CCSC2)C)CC)CC(C)(C)CN1C(=O)C(C)OC1CCCCC1 C1(NC(c2cc(CC)[nH]n2)=O)CC2CC(NC(c3ccn(C4CC4)n3)=O)CC2C1 Cc1cccc(C(=O)NC(C(=O)NCC(C)(CC)CO)c2ccco2)n1 C(=O)(C1CCCc2nn[nH]c21)NC1CC(OC)CN(C(c2c[nH]c(=N)o2)=O)C1 C1(NC(CSC)=O)CC(CNC(c2oc(C(F)(F)F)nc2C)=O)CC1O c1(OCCCC)ccc(N)c(C(=O)NC2CN(C(C3CCSC3)=O)CC2OC)c1 C12CN(CC13CC3)C2=O.C(C(=O)OCC1CC1)N(C(=O)OC)C.C(CCOC)NC c1(C(N2CCC(O)(CNC(c3occc3Cl)=O)C2)=O)cccc(F)c1C1CC1 C1(C(=O)NCC(C)CCCO)CCCN(C(c2cn(C(C)C)cn2)=O)CC1 C1(NC(C2(C)CC(C)=C(C)CC2)=O)CCC2CCN(C(c3cc(Cl)c[nH]3)=O)C1C2 c1(C(N(CCNC(C2(C)CC2C)=O)CC)=O)cc(Br)c2[nH]nnc2c1 c1(C(N(CCNC(c2ccc(C(C)C)o2)=O)C(C)C)=O)ccn2ccnc2n1 Cc1cc(Cl)cc(C(=O)NCC2(NC(c3ccc(SC4CC4)cc3)=O)CC2)c1O C(C(C(=O)N(C1CCCOC1)C)C(C)C)NC(C(COC)OC)=O c1(CC)ccc(C(C)=CC(=O)NC2CC(F)CN(C(C3CC(C)(O)C3)=O)C2)cc1 N1(C(C2C(OC)C2)=O)CC2(CCCN(C(=O)CC3CC3C(F)(F)F)C2)C1 C1(C(N2CC(C)C(NC(c3onc4c3CCCC4)=O)C2)=O)C2CCCCCCC12 c1(C(N)=O)cccc(C23CC2CNC3)n1 Cc1ccc(NC2CCN(C(=O)Cc3noc(C(C)C)n3)C(C)C2)cc1F C(=O)(C1CCCn2cnnc21)N1CCC(C)(NC(C2CCCCS2(=O)=O)=O)CC1 C1(=CC(=O)NCCC(CNC(C(C2CC2)OCC)=O)O)CN2CCC1CC2 C12(NC(C3(CC=C)CCCN3C(=O)CCN(C)C)=O)CCCN(CC1)C2 Cc1nc(C)c(-c2nc(C(C)C)nn2-c2cccc(C(F)(F)F)c2)o1 c1(C(=O)NCC2N(C(C3(C(C)(F)F)CC3)=O)CCC2)cc2c(cc1[N+](=O)[O-])OCO2 C(=O)(CC(CC)C(C)C)NC(CC(=O)N(CCC)CCN(C)C)C(F)F Cc1nc(Cl)ncc1NC(=O)CC12CCC1CN(C(=O)C1=C(Cl)CCC1)C2 c1(CC(C)C(=O)N2CCC2CNC(c2ccc(Cl)nc2O)=O)ccc(C#N)cc1 c1(OC(N)=O)ccc(Cl)cc1.C(=O)(C(CO)N)N(CC(=O)NCCC1(CO)CC1)C.CN CN1CCC(C(=O)N(C2CN(C(=O)Cc3cccc(C(N)=O)c3)C2)C)C1=O c1(C(N(CCCNC(C(CC)COC)=O)CC)=O)ccc(N)cc1F C1(NC(C(c2scc(C)n2)C)=O)(CNC(C2C(C)C2C)=O)CCOCC1 c1(NC2(CNC(CSCC#C)=O)CCCC2)nccc(C(N)=O)c1[N+](=O)[O-] C1(n2cc(CNC(c3cnn[nH]3)=O)nn2)CCCN(C(C23CCCCC2C3)=O)C1 c1(CC(=O)NC2(CNC(C=C(COC)C)=O)CCOC2)cn2c(C)csc2n1 CC1(CNC(C2(CNC(=O)CO)CCC2)=O)CCCCC1O C12(NC(C(=O)NCC)=O)CCCCCC1N(C(c1csc(C(F)F)c1)=O)CC2 c1(C(N2CCC(N(C(C3(CC#C)CC3)=O)C)CC2)=O)ccc(Br)nc1N n1(CC)nc(C(=O)N(CC(C)(C)NC(=O)C(C)Oc2cccnc2)C)c(C)n1 C1(C(=O)OC)C2CN(C(=O)CCC3(NC(C4CCCCC4O)=O)CCC3)CC12 c1(CC(C(=O)NCC(C)(C)NC(C(CC)O)=O)C)ccc(F)cc1 C1(NC(c2csc(-c3ccsc3)n2)=O)C=CCN(C(C2(Cl)CC2)=O)C1 N1(C(C(C)CC2CCCC2)=O)CCC(C)C1CNC(=O)C=CC1(C)COC1 c1(NC(c2ccccn2)C)cc(=NC(=O)CC2CCS(=O)(=O)C2)[nH][nH]1 C1(SC)COCC1NC(c1ccn(C)c1)c1nnnn1C N1(C(C(CC)(C)CC)=O)CCCC(C2CC2NC(=O)CC(C)c2ccco2)C1 CCCCC(C(=O)NCCc1ccc(F)cc1)NC(=O)CC1CSCCO1 C(=O)(C1CNS(=O)(=O)c2ccccc21)NCC(C)NC(C(CC=C)(C)N(C)C)=O C(=O)(C1=NN(CCO)C(=O)CC1)NCCCNC(=O)CC1(OCCO)CCOC1 C(=O)(C(O)CC(C)(C)C)NCC(c1cccc(OC)c1)NC(C1CCCS1)=O N1(C(C(CCCC)NC(C2CC(C3CC3)C2)=O)=O)CCC2(CNC(=O)N2)C1 c1(C(=O)NC2C(C(=O)Nc3c(OCCOC)cccc3)C2)cn2ccsc2n1 C(=O)(C1CCCc2c1ncn2C)NCC(CNC(Cc1n(C(C)C)cnn1)=O)O C(=O)(C(C)(C)CC(=O)NC(C1CCN(C(c2cnn(C)c2C)=O)CC1)C)OC C1(CC)CC(O)CN1C(=O)CC(C)CNC(C1CC(OC)C1)=O c1(NC(C2CC(F)(F)CN2Cc2ccccn2)=O)cc(F)c(F)c(F)c1 C1(CCNC(C(C)c2cc[nH]n2)=O)CN(C(=O)CCc2cn[nH]c2)CC1C C1(CNC(N2CC(CCO)C2)=O)CCOC(c2ccccc2)O1 N1(C(C=Cc2ccc(C)o2)=O)CCOCC(NC(=O)CN2CCCCC2C)C1 c1(C(=O)NCCC(C)NC(C2CC23CCC3)=O)csc2nccn12 Cc1c(C(=O)NC2CN(C(=O)CN3CC=CC3)CC2N=[N+]=[N-])nn2ccccc12 c1(C(=O)NC(CN(C(c2nocc2C)=O)CC)C)cc(C#N)cc(C)n1 C#CCCCCCCOC(c1cc(C(C)(C)C)ccc1OC)=O CCC(CC(=O)N1CC(CNC(C2(C#N)CC2)=O)C(C)C1)c1ccc(OC)cc1 OC1COc2cc(-c3ccc(CO)s3)nn2C1 CN1CCC(C)(CNC(C2(NC(c3ccc(C#N)s3)=O)CCCC2)=O)C1 CC(CC(C)(C)C)C(=O)N1CCCC(CNC(c2ccc(N)cc2[N+](=O)[O-])=O)C1 C(=O)(C(C)CC(N)=O)N1CCC(NCCNC(CCNC(=O)NC)=O)CC1 c1(C(=O)OC)ccc(C(=O)NNC(=O)OC)cc1 CC1CN(C(=O)C=CSCC(=O)O)C(c2ccc(Cl)cc2)CO1 C(=O)(C1=CCC(C)CC1)NCC1N(C(c2c(C)[nH]c(C#N)c2)=O)CC(O)C1O c1(C(=O)NCC(C2CCCC2)NC(CCC2CC(C)C2)=O)ccnc(C(N)=O)c1 C(=O)(C(F)(CNC(C1CN(C)CCO1)=O)C(C)C)NC1CCCC(C=C)C1 C(CO)(C(=O)NCC1(F)CN(C(=O)OC(C)(C)C)C1)N(C)C.C12CCN(C1)C2=O c1(OC)cc(O)ccc1NC(C1CC(O)CN1C(C1CCCS1)=O)=O C1(N(C(=O)CCc2nc(N(C)C)no2)CCC)CCCN(CCOC)C1 c1(C(=O)NCC(CCOC)NC(C2CC(C)=NO2)=O)ccc(CO)cc1 c1(C(N(CCCNC(c2cnn(C(F)F)c2)=O)C)=O)cccc(-n2ccnc2)c1 c1(CN(CCC(=O)NC23CCCC2C3)CCOC)cc(C)[nH]n1 Nc1nccnc1C(=O)NCC1CC(NC(C2CCC(C(=O)NCCO)C2)=O)C1 C1(C(=O)NCC2C=CC(NC(C(C(=O)OC)(C)F)=O)C2)Cc2nc(C)cn2C1 c1(NC2C(C)CN(C(=O)C3=CCCO3)CC2)ncc2ccnc-2[nH]1 CC(C(=O)N1CC(NC(c2ccc(CC3CCC3)cc2)=O)C1)C(C)n1cccn1 C1(NC(c2c(C)nc(C)o2)=O)CN(C(=O)Cc2cncnc2)CC12CCC2 CCCC(C(=O)NCC(C)NC(=O)CN1CC=CC1)NC(C)=O c1(NC(c2cc(COC)on2)=O)cccc(F)c1F CC1=NNC(=O)C1CC(=O)N(CCCOCCNC(=O)Cn1cccn1)C c1(OCCNC(=O)NC2CC(C(COCCF)O)C2)cccnc1 c1(OCC(=O)NC2(CCCNC(CC(C=C)C)=O)CC2)cc(F)cc(F)c1 Cc1cnc(C(N2CC3C(CNC(C45CCCCC4C5)=O)C3C2)=O)c(C)c1 CCCCCCC(C)C(=O)N1CCOCCC1C(=O)NCCC1CC(C)(C)C1 Cc1oc(C(=O)NCC2CCCC(NC(=O)Cc3ccnn3C)C2)cc1Br C1(CNC(C(C)n2cccn2)=O)CN(C(C2(C3CCC3)CC2)=O)CCCO1 c1(C(=O)NC(CCCCNC(C2CCC(CC)O2)=O)C)cccc(C)c1Cl c1(C(=O)NCC2CCC2NC(C2CCC(F)(F)C2)=O)cccc2oncc12 N1(C(C(C=C)OC)=O)CCOCC(CNC(=O)CN(C)C)C1 C1(CNC(CCC#C)=O)CCC12CCN(C(=O)Cc1cc(C)cc(F)c1)CC2 N1(CCC)CC(C(=O)NC(C)(C)CN2CCN(C(C3CC(=O)N3)=O)CC2)CC1=O C1(C(=O)NCC(CC)(C)NC(c2cnn(C)c2Cl)=O)CC2(CCOCC2)CO1 N1(C(c2n(CC#C)ccc2)=O)CC(CC(=O)NCC(C)OCC=C)CC1(C)C c1(NC(CC2CN(C(COCC(=O)OC)=O)C2)=O)ccc(C(F)(F)F)nc1C c1(C(=O)NCc2cn(C3CN(C(C(C)CN(C)C)=O)C3)nn2)ncc(Br)cc1O C1(S(C)(=O)=O)(C(N2CC(CNC(C3(C(C)C)CCC3)=O)OCC2)=O)CCC1 C1(C(=O)N(c2ccccn2)C2CC2)CCC(C)(C)C1.N12CC(C1)C(C)NC2=O Cc1cc(CCC(=O)N(C)CC2(CNC(C3C=CCCC3)=O)CC2)n(C)n1 c1(C(C2CC2)NC(C2N(C(C3(CN)CCCC3)=O)CCC2)=O)ccccc1F c1(-c2ccc(NC(Cc3c(C)cccc3)=O)cc2)ccc2[nH]c(C)c(C(N)=O)c2c1 CC1OC2(CNC(C3CCOC3)=O)CC1(NC(c1cccs1)=O)C2.O=C1CO1.CO C1(CC(=O)N(C(C=C)C)C)CN(C(=O)CSc2cn[nH]c2)CCO1 c1(CC(N2C(CNC(C(C)OCC=C)=O)CC(C)(C)C2)=O)nsc2ccccc12 C(=O)(CS(=O)C(F)(F)F)NCC(CC=C)NC(c1ccc2nccn2c1)=O N1(C(C=COCC)=O)CCC2(CC1)CC(C(=O)NCCC1CCCO1)CO2 Cc1nc(=N)[nH]cc1C(N1CCC2(CC2NC(=O)CNS(=O)(=O)N(C)C)C1)=O C1(NC(c2ccc(OC)c(F)c2)=O)CN(C(=O)CCNC(N)=O)CC2(CC2)C1 CC(C)CC(O)CNC(=O)C(CCOCCO)NC(C1OC2CCC1C2)=O N1(C(COCCC)=O)CCCC(NC(C2CCCC2C)=O)C1 c1(C(N2CCC(N(c3nnc(C4CC4)o3)C)C2)=O)cccc(-n2ccnc2)c1 N1(C(C2C(C)(C)CCCO2)=O)CCOC2CN(C(=O)C(F)CC3CCOC3)CC12 C1(C(=O)NC2CC(CC(=O)NCC(=O)OC(C)(C)C)C2)CC2CC(=O)CC(C1)C2 C12(C(N(CC(C)C#N)C)=O)CCC(CN(C(=O)CC3(C)CCOCC3)C1)C2 CCCCCCC(F)C(=O)N(C(C)CCNC(c1csc(C)n1)=O)C CC(C)C(F)(CNC(=O)COC1(C)CCC1)C(=O)NCCCN=[N+]=[N-] C1(C(N2C(C)C(NC(=O)CN3CCN(C)CC3)CC2)=O)CCn2cncc2C1 c1(N2CCC(C(=O)OCC)C2)nnc(-c2noc(C(C)C)n2)n1CC(C)C C(C)(C(=O)N1CCCCC1CNC(c1cc(C)nc(C)n1)=O)(C(C)C)NC(C)=O C(=O)(C1=CCCSC1)NCC=C1CCN(C(C(C2CCC(=O)CC2)F)=O)CC1 C1(S(=O)(=O)CC)(C(=O)OC(c2onc(CC)n2)C)CC1 c1(CC)ccc(C(=O)NCC2(C)CN(C(=O)Cc3ccoc3)CC2C)c(N)c1 CCCC(O)(CCC)CC(=O)NCCCNC(=O)C(CC)NC(=O)OC(C)(C)C.CC CCCCC(F)C(=O)N1CCCC(NC(c2sc(C)cc2C)=O)C1 C(=O)(CCP(C)(C)=O)N1C(CC(=O)N(C)Cc2cccnn2)CCC1 c1(C(=O)NCC2(F)CC(NC(C3(OC)CCOC3)=O)C2)ccncc1O C12(Cn3cc(CN(C)C4CC4)nn3)CC1CN(C(=O)CCC(=O)c1ccccn1)C2 C(=O)(CC(C(C)OC)NC(=O)CC1(CN(C)C)CCC1)N(CC(C)OC)C CP(C)(=O)C1(CNc2cn(C3CCOCC3)nc2C(C)(C)C)CC1 N1(C(C)C(=O)NC2CC(NC(=O)CO)CC2O)CS(=O)(=O)c2ccccc21 C1(NC(c2cc(OCC)no2)=O)CC2CC1CN(C(=O)Cc1ccns1)C2 Cc1c[nH]nc1C(=O)NC(C1CCN(C(c2csc(CC(F)(F)F)n2)=O)C1)C CS(=O)C1CN(C(=O)C=CCNC(=O)CC2CCCC(=O)C2)C1 C(=O)(CC1=CCCC1)N1CC(OC)C(NC(=O)Cc2cnccc2Cl)C1 C12(C(N3CCN(CCNC(=O)Cn4cc(Cl)cn4)CC3)=O)CCCN1CC(O)C2 c1(C(=O)NC2(CCCNC(CCOCC)=O)CC2)ccc(S(C)(=O)=O)o1 C1(C(N2CCC(C)(NC(c3ccc(NC)cn3)=O)CC2)=O)CCC12CCOCC2 c1(OC)c(C)nc[nH]c1=NCC1CCCC1NC(=O)C(C)Cc1ccncc1 Cc1cccc(C)c1C(=O)N(C(C)C(N1CC2CC2C2CC12)=O)C1CC1 CCC(C)C(CO)CN=c1ccnc(NCC2CCN(C(C)=O)CC2)[nH]1 C(C)(C(=O)NOCCC)=CCN(C(CCC)=O)C1CCC1 CCCC1C(=O)N1.c1(CSCCN)ncc(Br)cn1.C(=O)(OCC)OC C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1CC=C(CNC(CCC(=C)Cl)=O)CC1 c1(-c2ccc(C(=O)NCCN(CC(F)F)C)s2)cccc(Cl)c1 n1(CC)cc(CC(=O)NCc2c[nH]nc2C(=O)NC(CO)C2(O)CC2)cn1 C(=O)(C(C)C(C)(C)C)N(CCCCCNC(CCCc1onc(CC)n1)=O)CC C1(C(=O)NC(C2CN(C(=O)CCc3cn(C)nn3)CCO2)C)CCN(OC)CC1 c1(C(=O)NC2CC(CNC(C3CC(=O)C3)=O)C2)ccc2c(c1)OCO2 C1(C(C(=O)N(CC(C)CC2CCC2)C)OCC)CC(F)(F)C1.C1(C=O)(C(C)C)CC1 Cc1cc(Cl)ccc1COC(c1cc(CO)ccc1O)=O N12CCC(C)(CC1)C2=O.c1(C(=O)NCCOC)cc(N)ccc1C.C(CN)O c1(C(N(CC(C)NC(COC(CC)CC)=O)C)=O)c(C)noc1N N1(C(c2nccc(OC)n2)=O)CCC(S(=O)(=O)c2cccc(Br)c2)CC1 c1(C(=O)NC2CCN(C(C=C(COC)C)=O)C2(C)C)cnc2[nH]cncc1-2 c1(C(N2CC3CC(NC(c4cncnc4)=O)CC3C2)=O)n[nH]c2nccc(Cl)c12 C(=O)(CCc1ccon1)N(CCN(C(=O)CCC1CC1(C)C)C(C)C)C N1(C(Cc2cc(C)[nH]n2)=O)CCCCC1CC(=O)NC1CC1c1ccnn1C c1(C(=O)NC2CN(C(c3c(C)cc(C)o3)=O)CC2C)scc2c1OCCO2 N1(C(c2c(CC)ocn2)=O)CC2CC(NC(=O)CC3=CCCCC3)C(C2)C1 C(CC(C)(C)C(=O)NC(=O)C(C)C(F)F)OC.c12cn(nn1)CCS2 CC#CCCC(=O)N1CC=CC(NC(=O)C(C)Cc2ccc(COC)cc2)C1 c1(-n2c(NCC3CC4CCC3C4)nc(-c3ccccc3)n2)cccc2ncccc12 C(=O)(C(O)C(C)(C)C)N(CCC(=O)Nc1ccc(CO)cn1)C(C)C Cc1cccc(C(=O)NCC2CCCC2C(=O)NC2(CC(C)C)CC2)c1 C1(C(=O)NC(CN2CCCC2)CO)(NC(=O)Cc2cn[nH]c2)CC(F)C1 C1(COC(=O)CNC(=O)NC2CC2)CCCC(C(=O)Nc2ccccc2)CC1 Cc1cc(C)c(C(N2CCC(N(C)C(c3cc(Cl)nnc3O)=O)C2)=O)cc1N CC(C(F)C(=O)N(CCNC(=O)CCC(=O)c1cccnc1)C1CC1)C(F)(F)F c1(CSCCNC(C(=O)NC(c2nc(C)[nH]n2)C(C)C)=O)ccc(O)cc1 C(CCN=c1nc2[nH][nH]cc-2c(O)n1)NC(C1(C(F)(F)F)CCCCO1)=O N1(C(CC)=O)CC(C(=O)NCc2ccccc2OC)CCC1C C(C(C)C(=O)NC(C)(C)C(=O)N1CCCC1)(c1cccc(Br)c1)NC c1(C(=O)NC(CN(C(c2csc(C3CC3)n2)=O)CC)C)cc(N)ccc1[N+](=O)[O-] N1(C(c2cnc(OC)c(Cl)c2)=O)CCC2(C1)CN(C(c1c(Cl)cccc1Cl)=O)C2 c1(C(N2C(C(N(C)Cc3nnc(C)o3)=O)CC=CC2)=O)c[nH]c2nccc-2c1 c1(CC)sc(=N)[nH]c1C(=O)N(C(C)CCNC(C1CCN1C1CCCC1)=O)C C(C(COC)C(=O)NCCc1ocnc1CNC(C1CCC(F)CC1)=O)OC N1(C(C(C)CN(C)C(c2cnn3cccc3c2)=O)=O)CC2(CCC(=O)NC2)C1 N1(C(C(=O)NC(CC)C)CCC2CCOCC2)CCn2c(C)nnc2C1C N1(C(C=CC)=O)CCCC(N(CCO)C(c2cc(C)cs2)=O)C1 C(=O)(C1=CC2CCCC12)NC1CCC(COCC(=O)Nc2ccnc(OC)n2)C1 N1(CCC2OCC(C)(C)C2)CC(=O)N(CCC2CCC2(F)F)C1=O C1(C(N2CCC(CN(C)C(C3CCSCC3)=O)CC2)=O)CNC(=O)CC1(C)C CC1(C)CCOC(C(=O)NCCCCNC(C2CC2c2ccnn2C(C)C)=O)C1 C1(CC(=O)NCCN(C(C)C)C(c2ccc(=N)[nH]n2)=O)NC(=O)CNC1=O C1(CNC(c2c(OCC)n[nH]c2)=O)CCC2(CN(C(C3CCCO3)=O)C2)O1 c1(C(N2CC=CC(NC(C(COC)(F)F)=O)C2)=O)ccc(F)cc1OC N1(S(=O)(=O)CCNCc2ccccc2)CCC2(CCCCC2)CC1 CC(F)(F)C(C)(C)C(=O)NCCCNC(=O)CC1CCC2(CC1)COC2 C1(C)(CNC(c2nc(C(C)(C)C)oc2)=O)COCCN(C(=O)CC2COC(=O)C2)C1 c1(OC)ccc(C(N2CCC(C3CCCN3C(=O)CC(F)F)C2)=O)c(C)c1OC c1(C(=O)NCCCC(C)NC(C2CC2Br)=O)cc(C(F)F)n(C)n1 CC(F)(F)CCC(=O)NC1CC12CCN(C(C1CC(CC3CC3)C1)=O)C2 N1(C(C#CC(C)C)=O)CC2CC(NC(=O)CCc3nc4ccccc4s3)CC1C2 C1(CNC(CCCOCC=C)=O)CCN(c2nnc(-c3ccon3)s2)CC1C c1(C(=O)NCC2N(C(C=NOC)=O)CCC2C)cncc2sccc12 c1(C(=O)NC2CCCC(NC(CNS(CC)(=O)=O)=O)C2)cc(Cl)cc(C)c1C c1(C(=O)NC(CNC(C(CC)(C)OC)=O)CC(F)(F)F)cccc(F)c1C#N C1(NC(C(CC(C)C)NC(c2c(C)cns2)=O)=O)CC2(COCCO2)C1 c1(C(N2CC3CC3C2)=O)cccnc1NC(c1ncccc1C(=O)OCCO)=O C1(NC(CSCCC)=O)CC2CCC1C1CN(C(=O)C(C)C(C)C)CC21 Nc1cnccc1C(=O)NCC1(CNC(=O)C=CC(F)(F)F)CCCCC1 N1(C(C2(C)CCCO2)=O)CC2CC(O)C1C2NC(c1ccc(C(F)F)cn1)=O N1(C(CC(COC)NC(C2(N3CCCC3)CC2)=O)=O)CCCCC(CO)C1 c1(C(N2C(CNC(C3CC3C(F)F)=O)CCCC2)=O)cc2c(=O)[nH]ccn2n1 C#CC1(C(=O)NCCC2CCCCO2)CCN(C(c2n[nH]c(C)n2)=O)CC1 c1(C(=O)NCC2CC(NC(C(CC)CC3CCCCC3)=O)C2)nccc(Cl)c1C Cc1c(-n2nnnc2C(c2ccn(C(C)C)n2)NCC(C)(C)F)cccc1Cl N1(C(c2cnc(OCC)s2)=O)CCOCC(NC(=O)CCc2cccc(F)c2)C1 c1(OCC)ccc(CNc2nc(Cl)ccc2C(N2CCOCC2CO)=O)cc1I C(=O)(C(C)(O)C(C)C)N1C(CC(=O)NCc2cn(CC)nn2)SCC1 N1(C(COC(CC)C)=O)CCOC2(CCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)C1 c1(C(=O)NC)cc(C(C)C)[nH]c1CC(CCNC(C(CC)CC(=O)OC)=O)OC c1(NCC(C2CCOC2)NC(=O)Cc2cnns2)ncc(Br)cn1 c1(CN(C(CN(c2cccs2)C)=O)C)ncc[nH]1 c1(-c2c(CN3C(C(=O)O)CCCC3)nccc2)ccc2ncsc2c1 C1(=CC(=O)NCC2CCN(C(C3CCO3)=O)C2)CCOc2ccccc21 C1(C(=O)NCC23N(C(CCC(C)=O)=O)CC(CC)(C2)C3)CCc2nncn2CC1 C(C(C)(Cn1cccn1)NC(C12COC(C1)C2)=O)NC(C=C(COC)C)=O CN1C(=O)C(C(N2CCCC(CCNC(=O)C(C)(C)O)C2)=O)Cc2ccccc21 C12CCCN(CC1)C(=O)C1(CC1)C(=O)N2C.c1(C)ccnc(Cl)c1.N(C)C c1(C(=O)NCCCOCCCN(C2CCC2)C)cc2scnc2[nH]1.C1(=O)CN1 C1(NC(c2ccc(C)cc2C)=O)CCN(C(C2CC3CCC(C2)C3)=O)CC1(C)C C(C(C)(C(C)C)NC(=O)Cn1cccn1)NC(C1(OC)CCC1)=O c1(CNC(=O)NC(C2CCCCC2)(C)C)ccnc(Cl)c1 c1(C(N(C)CC2CCCCN2C(C2(CO)CCCO2)=O)=O)ncc(Cl)cc1Cl c1(C(=O)NC(CC)C(=O)N2CCC2CNC)ccc(C(=O)N(C)C)cc1 C1(C(=O)NCC2(NC(=O)C(C3CCOCC3)F)CCC2)CCC2(CC1)CC2(F)F CC(C(=O)N(CCNC(=O)C#CC1CC1)CC1CC1)C(F)(F)F Cc1cc(C(=O)NCC2CCCN2C(c2cccnc2Cl)=O)cc(O)c1 c1(C(=O)NC2CN(C(C3CC(O)C3)=O)CC2CC2CC2)cc(O)ncc1Br N1(C(=O)CC2CC=CCC2)CCCN(C(C2CC(F)(F)C2)=O)C(CO)C1 c1(C(=O)NCC2(F)CN(C(=O)CCOCC3CCC3)C2)cc2n(c1)CCCC2 c1(C(=O)NC(CCOCC)C)cnn(C)c1I NC1CN(C(C2CCCC3CCC23)=O)CC2(CC2)C1 C1(NC(C(C=C)c2ccccc2)=O)CCN(C(c2sncc2CC)=O)CC(O)C1 CN1CCOCC1C(N1CCC(CO)(NC(=O)CCOCC2CCC2)C1)=O c1(OC)ccc(OC)c(C(=O)NCCN(C)C(c2ccc(O)nc2Cl)=O)c1 CCC(O)C(C)(C)C(=O)NCCc1c(C)cccc1F CC(CC(C)(C)C)C(=O)NCC1CN(C(c2cc(C3CCC3)no2)=O)CC1(C)C N1(CC(=O)NC2(CN(C)C(C34CC(F)C3C4)=O)CC2)C(=O)NC(C)(C)C1=O C1(N(C(C=CC=CCC)=O)C)CN(C(=O)C=Cc2cccc(CO)c2)CC12CC2 N1(C(CCCCCOC)=O)CC(C)CN(C(C2OC(C)CC2C)=O)CC1C C1(C(=O)NCC(C(C)C)NC(=O)CC#N)CCCCN1Cc1ccccc1 C(CCCS(C)(=O)=O)NC(C(=O)N(C)Cc1ncn(C)n1)=O CC1CC(=O)NC(C(=O)N(C)CC2(C(=O)NOCCCF)CC2)C1 N1(C(C(C)(C2CCOCC2)OC)=O)CCOC(CCNC(=O)CC2CN(C)C2)C1 C1(NC(=O)OC(C)(C)C)CCC(C(=O)NCCN(C(=O)CC23CCCC2C3)C)CC1 CC1C(NC(=O)CC(C2CC2)C2CC2)CCCN1C(=O)Cc1ccccc1 C(=O)(C(C)(C)C(C)NC(=O)CSCC)NC(CC)CC(C)C C1(CSc2ccn(C)n2)CCC2(CN(C(=O)C(F)CC3CCC3)C2)O1.C1C(=O)N1 c1(C(=O)NC(C=CC(=O)NC(C)C)C)cccc(CNC2CCC2)c1 C12(C(=O)NC(CCCC)CO)CCN(C(=O)CCc3ccncn3)CCC1C2 CCCCCCC(CC)NC(C12C(NC(c3cn(C)cn3)=O)C3CC1C2C3)=O CC1=NNC(=O)C1CC(N1CCC(C(=O)N(C)CC2CCCC2O)C1)=O C1(CC)(NC(=O)C(C)=C(C)C)CCCN(C(c2ccncc2OC)=O)C1 c1(C(N2C3CN(C(CS(=O)(=O)NC)=O)C(C3)C2)=O)cc(N)c(C)c([N+](=O)[O-])c1 C(C(C(=O)NC(c1n[nH]c(CC)n1)C)NC(=O)CC1CCCOC1)SCC N1(C(C2N(C(CCCN(C(C)=O)C)=O)CC2)=O)CCCC1(C)CC(C)C c1(C(N2CCNCCC3(NC(C=CSC)=O)C(C2)C3)=O)cc2ccc(F)cc2o1 N1(C(C(CNC(c2cccc3c2CCC3)=O)O)=O)CCC2(C=CCO2)C1 N1(C(CC(C)n2cccn2)=O)CCCC(O)(CNC(C2CCC3(CCC3)O2)=O)C1 C1(C(=O)NCc2ccc(Cl)cn2)CCNC2(CC2)C1.c12cccc(c1)OC2 C1(CC(=O)NCC(CCOC)NC(CCCC#C)=O)CC2CCC(C1)N2C C(=O)(CCC(=O)NC1(CNC(c2c(Cl)cnn2CC)=O)CCC1)N(CCC)CCC n1(CC)nc(C(=O)NCC(CC(C)C)NC(c2cccc(C(F)F)n2)=O)c(C)n1 C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCc2c(nc(C(C)(C)C)s2)C1 CC(C)(CC#N)C(=O)NCC1(F)CCC(NC(=O)CCc2ccc(F)cc2)C1 Cc1ccc(C(=O)NCC(C)NC(=O)Cc2cnn(C(C)C)c2)c(N)c1C Cc1cc(=NC(=O)C2CCN(C(C3CCO3)=O)C2)[nH]n1C c1(C(=O)NCCN(C(c2c(Cl)c(C)n(C)n2)=O)C)cn2c(n1)CCCC2C C(C1CC1)(C1CC1)=CC(=O)NCCC(C)N(C(=O)C(O)C1CCCC1)C C(CC(=O)N(C)Cc1ccns1)(CC(C)C)NC(c1c(C)cc(N)cn1)=O c1(C(=O)NC(CC)(CNC(C2CC2C2CCCO2)=O)CC)cnc(O)c(Cl)c1 C(=O)(CCNC(=O)NC1CCCO1)NCC1C(NC(C2CCC2)=O)C1 CC1CC=C(C(=O)NC2CC(O)(CNC(c3cc(C(F)F)n(C)n3)=O)C2)CC1 c1(C(C(=O)NC2CCN(C(C3(CC)CCCCO3)=O)C2)O)cc(F)cc(F)c1 C1(C(C(=O)NCCOC)NC(=O)NCCc2ccncc2)CCC(N(C)C)CC1 C1(CNC(c2c(CNC(C3CN(CC)C(=O)C3)=O)occ2)=O)CC(C2CC2)=NO1 c1(OC)ccc(N2CC(C(=O)NC3CCC3NC(C3CCO3)=O)CC2=O)cc1Cl N1(C(c2c[nH]c(=NC)o2)=O)CCC(NC(c2nn(C)cc2SC)=O)CC(O)C1 C(=O)(CC(C)(C)O)N(CCNC(CCCN(C(C)=O)C)=O)C1CC1 Cc1cc(C(=O)NC(C(=O)NCC(C)(O)CCO)C2CCC2)nc(C)n1 n1(CC(=O)N(C2CCN(C(C3(C#N)CC(C)C3)=O)CC2)CC#C)ncccc1=O C1(CC(N)=O)(NC(c2c(C)cnnc2)=O)CCN(C(C2(n3nccn3)CC2)=O)CC1 C1(C)(NC(c2c(C)nn(C)c2)=O)CCCN(C(=O)C(n2cc(Br)cn2)C)C1 C1(CNC(c2cccc(C(F)F)c2)=O)CN(C(=O)Cc2ccccc2Br)CC1O c1(CN2CCC(NC(c3cc(C)n(C)c3)=O)C(O)C2)cc2ccccc2nc1O c1(C(=O)NCC(C)OC)nc2ccc(-c3ccc(F)cc3SC)cc2o1 N#Cc1csc(C(=O)NC2CCCC2NC(=O)C=CC(F)(F)F)c1 N1(C(C2(CC=C)CC2)=O)CCC(NC(=O)C2=CC(C)(C)C2)CC1C CC(=O)CC(C)(C)C(=O)NCC=CC(=O)NC1CCC(CCO)CC1 Cc1cc(C(N2CCN(C(=O)Cc3coc(C(F)F)n3)C(CO)C2)=O)nnc1C C[S+](C)CCC(O)C(=O)NC1(CNC(=O)C(C)(C)C)CC1 C1(NC(C(N2CC(OCCOC)C2)=O)=O)CCC(F)CC1 C1(CNC(COC)=O)CN(C(c2c(C)ncn2O)=O)CC12CCC2 c1(C(=O)NC2C(NC(C(CC#C)O)=O)COC2)cc2cc(Br)cc(C)c2[nH]1 C=CC(C)(O)CC(=O)N1CC(F)CC1C(N1CCC1COC)=O N1(C(C2C(=C)C2)=O)CC(O)(CCC(=O)NCCC2(C)CCOC2)C1 C1(C)(C(N2C(CNC(C3CC4CC4C3)=O)CC(OC)C2)=O)COC(=O)OC1 c1(C(=O)NC(c2cn(-c3cccs3)nn2)C)ccc(-c2cccs2)nc1O c1(CNC(CC2C(C)CCCC2)=O)nn(C)c2c1CN(C(=O)Cn1cncn1)CC2 C(=O)(CC1=NNC(=O)C1)NCC(CCC)NC(c1ccc(Br)c(O)n1)=O c1(C(CN(CC(C)C)C(=O)CNC=O)C)ccccc1Cl c1(C(=O)NC2CC(NC(C3C(C)OC(C)C3)=O)C2)cnc2[nH]ncc2c1 c1(C(O)CN2CCN(Cc3ccco3)CC2)ccccc1Cl Cc1cc(=O)cc(CNC(c2conc2CNC(C2CC2(C)C)=O)=O)[nH]1 C1(c2cn(CCC=C=C)nn2)C(C)CCN1C(c1ccncc1CC)=O C1(C(=O)NC(CCCC)(C)C)C2CC3C(C2NC(C2CCC(=O)NC2)=O)C13 N1(C(c2cnccn2)C(=O)NCCOC)CCN(CCCF)CC1 c1(CCC(=O)NCC2C(NC(Cc3nnc(C)o3)=O)C2)c(F)cccc1Cl C=CCCCC(C)(C)C(=O)NCC(O)CNC(c1cccc(CSC)c1)=O C1(C(=O)NCC=CCNC(=O)C(F)C(F)(F)F)CC2(CCCC2)CO1 O=C(C1=CCCCCC1)NCC1(C(=O)NC23CC2COC32CCC2)CC1 N1(C(=O)CCC(F)(F)F)CCC2CCCN(C(c3ccnc(C(F)F)c3)=O)C2C1 CC(O)(C(=O)NC1CCCCCN(C(=O)CCn2cnnn2)C1)C(F)(F)F N1(C(c2ccc(C(C)C)o2)=O)CC(C)(C)CC1CNC(c1cc(C2CC2)n[nH]1)=O Cc1scc(C(N2CCN(CC(=O)NC3CCCC3C(C)C)CC2)=O)c1C CCS(=O)(=O)CCCNC(N1CCN(c2ccc(N(C)C)cc2)CC1)=O C=CCC(C)(CC=C)NC(C1CCN(C(C2CCC(=O)O2)=O)CC1)=O c1(C(N2CCC(N(C(CCCOCC=C)=O)CCC)C2)=O)cccc2ncoc12 C1(CNC(C(C)C#N)=O)CN(C(=O)C(C)(C)n2cc(Cl)cn2)CC1N(C)C c1(C(=O)NC2C(CNC(CCNC(N)=O)=O)CCCC2)ccnc(O)c1F C1(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CCCN(C(=O)CC2(O)CC2)C1 Cc1nncn1NC(=O)C1CC(CNC(=O)CCOCCN(C)C)C1 c1(SCC(N2CC(C)C(NC(C3CC4(CC4)C3)=O)CC2)=O)nc2ccccc2[nH]1 Cc1ccc2oc(C(=O)NCC(C)NC(c3cc4cc(Cl)ccc4o3)=O)cc2n1 C=CCC(C)(C)CC(=O)N(C1CC(NC(c2cnc(O)c(F)c2)=O)C1)C c1(N2CCC(CN(C(=O)CCC3CC(F)(F)C3)C)CC2)ccn2nccc2n1 CC1C(NC(C23CC2C3)=O)C(C)CCN1c1ccnc(C2CC2)n1 c1(OCC(=O)NCC2C=CC(NC(C(C)CC3CC3)=O)C2)ccccc1[N+](=O)[O-] C1(NC(C(C)(C)F)=O)CC2CC(C1)N(C(c1ccc(CC3CC3)cc1)=O)C2 N1(C(=O)C2=COCCC2)CCC2(CCN(C(c3ccc4c(c3)CCC4)=O)C2)C1 c1(C(N(C)CC2(NC(=O)C3=CCSC3)CC2)=O)cn2cnnc2cn1 N1(CC#C)CCCC1C(=O)N(C)CCOCCN.C1(C#N)(O)CC1 C1(NC(C2(C#C)CC2)=O)CCN(C(c2cc(C(F)(F)F)n[nH]2)=O)C(C2CC2)C1 Cc1ccc2nonc2c1S(=O)(=O)N1CCN2CCCC2C1 C=Cc1cncc(C(N2CCC(CC(=O)NC3CC(=O)N(CC)C3)C(C)C2)=O)c1 N1(C(CCCN(C(=O)CSCC(N)=O)C)=O)CCNC(=O)C1CCO N1(C(C(C)OCC#C)=O)CCCCC1CCCN(C)C c1(C(N2CC(OCCC)C2)C(=O)NCCCF)nn(C(=O)OC)nc1Br c1(C(=O)NCCN(C(C=CC(C)C)=O)C(C)C)cc(=O)c2ccncc2o1 c1(C(=O)NCC2(F)CC(CNC(c3cc(CC)no3)=O)C2)ccc(F)cc1C C1(C)(N(c2cc(NC(C)Cc3ccccn3)ncn2)C)CCS(=O)(=O)C1 CCC(CC(=O)N1CCCC1C1(C(N2CCNC(=O)C2)=O)CC1)C(F)F Cc1cccc(C(F)(F)C(=O)N(C2CCC2(C)C)C)c1 C#Cc1cc(C(=O)NCC2C3CCC(C3)N2C(=O)Cc2c[nH]nc2O)cc(F)c1 CCCC(C)(C)CC(=O)OC.N12C(=O)NC(C1=O)c1cccc(c1)C(=O)NCC2 c1(C(=O)NC(C2CC(NC(C3CCSCC3)=O)C2)C)ccnc(C(C)(F)F)c1 C(=O)(CCCCC(=O)NC(C1CCCN1C(=O)C(c1cn(C)nc1C)C)C)OC C12(C(=O)NCCNC(C(C)NC(C)(C)C)=O)CC(CO1)C2 C1(c2n(C(C)C)ncc2)NC(=O)CCC1NCc1c(Cl)nsc1Cl c1(CC)c(C)sc(NC(C2(C)CCC(NCc3csc(C)n3)C2)=O)c1C(N)=O C1(CNC(C(n2cnc(C#N)n2)C)=O)CN(C(=O)COc2ccccc2)CC1O c1(C(=O)NCC2C3N(C(C=CS(C)=O)=O)C(CC3)C2)cc([N+](=O)[O-])cnc1O c1(C(N2CC3CCN(C(COC)=O)CC32)=O)cncc2nc(C(F)(F)F)[nH]c12 CCC(CC(C)CO)NC(=O)C(=O)N(C)CCN1CCC(C)CC1 c1(CC(=O)NCC2C(NC(c3c(C)nco3)=O)CC2)ccc(NC(C)C)cc1 c1(C(N(CC(C)O)CCNC(C23CC(F)C2C3)=O)=O)cc(C(F)F)n(C)n1 C1(NC(CC(COC)(C)C)=O)CCCCCN(C(=O)C(C)OCCC(C)C)C1 N1(C(c2cnn(C(C)C)c2N)=O)CCN(C(=O)CN2CCP(C)(=O)CC2)C(C)C1 N(C1CCCn2ncnc21)C(C1(C(C)NC(=O)CCCCC#N)CC1)=O CCCCC(CC)C(=O)NCC1(CNC(C2CC23CC(C)(C)C3)=O)CC1 N1(C(CC(CC)CC)C(=O)NCCCOC)CCC2(CC1)CC2(F)Br c1(C(=O)NCCC2CCN(C(C(C)OC)=O)CC2)ccc2[nH]c(=N)oc2c1 C(=O)(CCC(=O)N1CCC(CC(=O)NCCN2CCOC2=O)CC1)OC(C)(C)C N1(C(c2ccc(OC)cn2)=O)CCC2(CC1)OCCC2NC(c1ccccn1)=O c1(C(N2CC3=C(C2)CN(C(C2CC24CC(O)C4)=O)C3)=O)nc2ccccc2[nH]1 c1(OC)ccnc(C(c2nnnn2C2CC2)NCc2cnccc2C)c1 N1(C(C(CN(C)C)(C)C)=O)CCC2(C1)CN(C(=O)CC1COC(C)(C)CO1)C2 N1(C(Cc2c(C)con2)=O)CCC(NC(c2cnc(Cl)cc2Cl)=O)C(C)C1 CC1CC(NC(=O)CC2CC3CC3C2)CCN1C(=O)COCc1ccnc(O)c1 CC1=C(C(=O)NCC2CCN2C(=O)Cn2nccn2)CCO1 C1(N)(C(=O)NCC(=O)NCCN(CCOC)Cc2ccco2)CCOCC12CCC2 CN(C)S(=O)(=NS(=O)(=O)Nc1c(Cl)cc(C=CC)cc1CCC1(CC)CC1)c1ccccc1 c1(C)ccc(OC)cc1.n1(SCC)ccnc1CC(=O)NCC1CCCC1.C12(CC1)CN2 C1(NC(C(C)OCCC=C)=O)CCC(O)CN(C(c2ccncc2)=O)C1 Cc1ccc(OCCC(=O)NC(C)C(C)(C)NC(C2C=CCC2)=O)cc1 Cc1csc2ncc(C(=O)NCC3CC4(CC4)CN3C(=O)CC(O)CN(C)C)n12 c1(C(N2CCC(C(=O)NCCN(C)CC3CCC3)CC2)=O)cc(F)cc(N)c1F c1(CNCC2(SC(C)C)CCCCC2)ccc(Oc2ccccc2)c(C#N)c1 C1(CNC(c2n(C)c3c(c2)ccs3)=O)CC2CCCCC2N1C(C1CCO1)=O C12COC(C1)CNC2=O.C1(CC(=O)CC=CCl)COC(CNC(=O)C2CC2)C1 n1(CC(=O)NC(CNc2nc[nH]c3nccc2-3)C2CC2)ccc2nc(O)nc(O)c12 C1(CNC(CC2C(C)(C)C2)=O)N(C(C2CC3(CCCC3)C2)=O)CCCC1(C)C C1(NC(Cc2c(C)noc2)=O)CC(CO)N(C(c2ncc(Br)cn2)=O)C1 C1(NC(CC(C)C)=O)CC(C)N(C(c2cnc(OC(C)C)cn2)=O)C1 Cc1ccnc(C(=O)NCC2CCC(NC(c3cnns3)=O)C2)n1 Cc1nc2ccc(C(N3CC(NC(=O)CSC(F)(F)F)CC(C)(C)C3)=O)cn2n1 Cc1cc([N+](=O)[O-])cc(C(=O)NCC2N(C(c3cnco3)=O)CCCC2(C)C)n1 Cn1nnc2cc(C(N3CCCOC(CNC(C4CCC4(F)F)=O)C3)=O)sc12 c1(C(N2CC3(CC(NC(CCOC)=O)C3)C2)=O)sccc1S(=O)(=O)C1CC1 c1(OC)cc2c(cc1C(=O)NC1(C)CCCN(CCc3ccccc3)C1)CCC2 N1(C(C)=O)CCOCC1C(=O)NC(C)CC1CN(C(c2coc(N(C)C)n2)=O)C1 Cc1noc(-c2cn(CCCC(=O)N(C3CCCC3N(C)C)C)nn2)n1 C=CC(O)C(=O)NCCCOCCOCCNC(C1(CC=C)CCOC1)=O N1(C(C(C)(C2CC2)OC)=O)CC2(CCCC(CNC(c3cnn(C)n3)=O)O2)C1 CC1C(=O)N2CCN12.C1(C[SH](=O)=O)C2CCOCC12 CC1COc2ccccc2CN1C(c1cccc(C(F)F)c1F)=O c1(OC)c(NC(c2nc(-c3cc(O)cc(O)c3)sc2C)=O)cccc1Br C1(C(C)C)COCCN(C(C2CC(NC(=O)CCOCC(C)(C)C)C2(C)C)=O)C1 C1(CC(=O)N(CC(CC)C)C)CCN(C(C2C=CCCC2)=O)C1 C(=O)(C(F)C(C)CC(C)(C)C)N1CCC(C)(NC(CN(C(=O)OCC)C)=O)C1 C(=O)(C1CCc2nccn21)N1CC(F)(CN(C(C2CCc3cnnn3C2)=O)C)C1 N1(C(C(c2ccn(C)c2)C)=O)CC2(CCN(C(c3cnc4c[nH]nc4c3)=O)C2)C1 Cc1cc(F)c(C(=O)N(C)CC2(NC(=O)CCCOC(C)(C)C)CC2)cc1F N1(C(CCCC=C)=O)CCCCC2(C1)CN(C(c1ccc3nc(S)oc3c1)=O)C2 C(CCC(=O)N(C1CC1)CC1CCOC1)(C(C)C)NC(C(CCC)=CCC)=O N1(C(CCc2nc(=N)[nH][nH]2)=O)CC2CC2(CNC(C2C3CNC(=O)C23)=O)C1 c1(C(=O)NC2C(CNC(c3cnnc(C4CC4)c3)=O)C2)cccc2ccnn12 c1(CNC(N2CC(Cn3cc(I)cn3)C2)=O)nnc2n1CCS2 CCCC(C(=O)OC)C(=O)N1CCCN(C(=O)Cc2cc(C)on2)CC1 Cc1snnc1C(=O)NC1(C)CC(NC(=O)CCN(C(C2CCCO2)=O)C2CC2)C1 CN1CCC(C(=O)NCCCC2CCCN2C(C2CC(O)C2)=O)c2ccccc21 C(C(O)C(F)(F)F)N(C(=O)CN(C(=O)Cn1cncn1)C1CC1)CC1CC1 C(C)(CCC(=O)N1CC(NC(c2cn(CCF)nn2)=O)C1)OC N1(C(C(C)(CO)OC)=O)CC2CC(C1)C(CO)C2NC(C1(C(C)C)CCC1)=O c1(CC(=O)NCC(CNC(CC(C=C)(C)O)=O)O)csc2c(Cl)cccc12 N1(C(c2c(C)occ2)=O)CCOC2(C1)CN(C(=O)C(C)OC1CCCC1)C2 C(=O)(C1COc2cc(C)c(C)cc21)N(CCNC(=O)CCc1nncs1)CC N1(C(COCC=C)=O)CCOCCC1C(=O)N(C1CC1(C)C)C c1(CC(=O)NCC(C(C)(C)C)NC(=O)Cn2cccn2)nc2c([nH]1)CCCC2 C1(CCC=C)(C(N2CC(N3CC(O)C3)C2)=O)CN(C(=O)C(C)Cn2cccn2)C1 C12CC3CC3N1C2=O.C12(CNC(CCOC(C)C)=O)COCC(C1)C2 Cc1ccc(C(N2CCC(C(C)NC(C3CC(C)OC3C)=O)C2)=O)nc1 Cc1c(C(=O)NCC2C(C)CCN2C(=O)CNS(N)(=O)=O)c(C(F)(F)F)nn1C C(=O)(CCCCCF)N1C(CC)C(C(=O)NCC(O)CC(=O)OC)CC1 C1(C)(C(=O)NCC2COCCN(C(CC3CC(OC)C3)=O)C2)CCC(C)=C(C)C1 C1(NC(c2ccc(CC)cc2)=O)CC2CCC1(NC(c1cnc3n1CCC3)=O)C2 C1(C(=O)NC2CCC(N(C)C(C3C(C)C3C)=O)C2)(NC(N)=O)CCC(F)(F)CC1 c1(C(=O)OC(C)(C)C)ccccc1CNC(=O)Cc1ccc(-n2cccc2)cc1 c1(CC)ccc(CNC2CCC(CNC(c3cc(F)cc(F)c3)=O)CC2)c(O)c1 C(=O)(C(C(C)O)NC(=O)C(C)O)NCCCNC(C)=O N1(CCC(=O)NC(C2CCCSC2)COC)C(=O)c2ccccc2C1=O c1(NC(C2N(C(Cc3ccc(C)nc3)=O)CC(F)(F)C2)=O)ccn2nccc2c1 C(=O)(CCCCC(C)C)N1CC2CC(CNC(C(c3ccccc3)SC)=O)C2C1 C(CCC(=O)NC1CC(C(F)C(=O)NCCS(C)(=N)=O)C1)OCCOC CCC(c1ccccc1)=CC(=O)NCCC(O)CNC(c1cnns1)=O N#Cc1cccc(C(CF)NCC2CCC3(COC3)C2)c1 Cc1ccc(Cl)c(C(=O)NC(CNC(c2cn(C)nc2Cl)=O)C2CC2)c1N c1(CNC(c2ccccc2)COC(C(=O)N(C)C)=O)ccc(C2(CN)CC2)cc1 Cc1ccc(C)c(C(=O)NC(C(=O)NC2(CO)CC3(CCC3)C2)c2cccs2)n1 CC1CN(C(c2ccccc2NC(N)=O)=O)CC(C)N(C(=O)C2CC2)C1 C1(C(=O)NC(C2CCCC2)CNC(=O)CC2CC2(F)F)CC(F)(CO)C1 C(CC(C)(C)CC(=O)NC1COCCN(C(=O)CCc2scnc2C)C1)OC S(=O)(=O)(C1CC1)NCC(N1CC(O)(CNC(c2csc(Cl)n2)=O)C1)=O C1(N(C(=O)CC2CC2C(C)(C)C)C)CC12CCOC2.N12CCCC1(C)CNC2=O C1(NC(c2cccn(C)c2=O)=O)CCC2(CC1)CN(C(=O)C=Cc1ccsc1)C2 C(N=c1ccn2nccc2[nH]1)C1CCCN(C(C2CCCN(c3nncs3)C2)=O)C1 C(=O)(C(CNC(=O)C(C)COC)C(C)C)NCC(C)OCC#C CC1CCN(C(C2CSCN2C(=O)C=Cc2cscn2)=O)CCS1 n1(CC(=O)NCC2CCCO2)cc(C2CC2)cn1.O=C1C(=O)NC2CC(C2)N1 CC1CCCCC1(CN(C(=S)Nc1cccc(Br)c1)C)OC(F)F CC(C)C(C(=O)N1CCC(CCO)C1)C(C)OCC(=O)NCc1nc[nH]n1 C12(NC(=O)C(CC3CC3)c3ccccc3)CC1CN(C(c1cc(CO)on1)=O)C2 c1(CC)ccc(Cl)c(C(=O)NC2CN(C(C3CCOC3)=O)CC23CC3)c1 c1(CC(=O)OC)cc(NC(c2nn(-c3ccccc3F)cc2C)=O)c(O)cc1F Cc1cc(-c2noc(CC3ON=C(C(=O)OCC4CC4)C3)n2)ccc1O c1(OC)nc(C)ccc1C(=O)NCC12CC(CN1C(c1csc(C)c1N)=O)C2 c1(C(N2C(CNC(Cc3cc(CC)no3)=O)C=CC2)=O)nc(Br)cnc1N c1(NC(CC(N2CC3(CN(C(CC)=O)C3)C2)=O)=O)ccc([N+](=O)[O-])cc1CNC c1(N)ccc(C(=O)OC)c(C)c1.C1(C(N(c2n(CC)nnn2)C)=O)(CF)CCOCC1 C(=O)(CC(C)C(=O)NCC1CCC(C(=O)N(C2CC2(C)C)C)CC1)OCC Cc1ccc2sc(N(C(C)CCNC(c3ccc(N=[N+]=[N-])c(C)c3)=O)C)nc2c1 c1(NC(C)C(C2CCOCC2)C)ccc(S(=O)(=O)N(C)Cc2ccccc2)cn1 C1(N(C(CCCNC(CN(C(=O)OCC)C)=O)=O)C)CC(C(=O)OC)C1(C)C c1(C(=O)NCC2CCN2C(C2CC(C3CC3)=NO2)=O)cc2c(cc1[N+](=O)[O-])OCO2 N1(C(C)=O)CCCCC1C(=O)NC(C)CNC(c1ccnn1C1CC1(F)F)=O c1(N2CCC(NC(C)=O)CC2C)ccc([N+](=O)[O-])c(C#N)c1 c1(C(=O)NC2CC3(CC(CNC(=O)C=CC(F)(F)F)C3)C2)noc2ccccc12 c1(OCC=C(C)C)ccc(Br)cc1CC1C=CCCC1 N1(C(=O)CSC2CCCCO2)CC(NC(C2(CO)CCC2)=O)CC12CCC2 Cc1nn(C)c(F)c1C(=O)NC12CCOC(CNC(=O)CC(C)N(C)C)(C1)C2 c1(C(=O)NC(C)(CNC(c2cc(CF)on2)=O)CO)[nH]c2ccccc2c1Br N1(C(c2c(CC)c[nH]c2)=O)CCCC1(C)CNC(=O)CC(=O)NC1CC1 N1(C(CCOCCOC)=O)CCN(C(c2ncc(Cl)cc2F)=O)CC(C)(F)C1 Cc1c(C(N2CCC(C(C)NC(=O)C(Cl)=CCl)C2)=O)ccc(F)c1F Cc1nc2nccc(C(=O)NCC(C3CC3)NC(=O)C(C)S(N)(=O)=O)n2n1 C(=O)(C(C)(C)CC(=O)NCC1CC(O)CN1C(c1nccc(OC)c1C)=O)OC CCC(C)(C(=O)NCC(C)(C1CC1)NC(C1CCC(C(C)C)CC1)=O)OC c1(C(=O)NCCN2CCN(C(CCC(=C)Cl)=O)CC2)cc(S(N)(=O)=O)c[nH]1 Cc1cc(C(N)=O)n(C(C)(C)Cc2cn(C(C)CNC(c3cnc(O)[nH]3)=O)nn2)n1 C12(CNC(C3(C)CC4CC4C3)=O)CCC(CC1)N2C(=O)CCCCNC(N)=O C1(N(C(=O)CCc2cccs2)C)CCCN(C(C2CC2C#N)=O)CC1 C1(NC(=O)C(F)n2cccn2)COC2(CCN(C(C3(C(N)=O)CC3)=O)CC2)C1 c1(C(=O)NC2C(NC(CC3N(CC)CCC3)=O)CCC2)c(Br)ncn1C C#Cc1cn(C)nc1C(N1CCC1C(=O)N(C1CCOCC1C)C1CC1)=O c1(OCC)ccc(C(=O)NCC2(O)CN(C(=O)CC3CCCC3(F)F)C2)cc1C c1(C(C)=O)ccc(C(=O)N(C2CCC(CNC(C3CCCN3C)=O)CC2)C)cn1 CCC(C)(C(=O)NCC1(F)CC(CNC(C2(C)CCCS2)=O)C1)C(N)=O C1(NC(Cc2cc(CC)no2)=O)CCN(C(=O)C=Cc2ccccc2Cl)C1(C)C C12(C(=O)NCC(CC)NC(c3cscc3C(N)=O)=O)CCC(CC1)OC2 N1(C(C2(CCC)CCC2)=O)CCCN(C(c2ccc(Cl)c(F)c2)=O)CC1CO Cn1ccc2ccc(C(N3CCC(NC(=O)Cc4nc(=N)[nH][nH]4)C3)=O)cc12 C1(C(=O)NOCCOCc2ccccc2)CCN(C(=O)c2coc(CO)c2)O1 c1(NC(C(C2CN(C(C3CCC(CC)O3)=O)C2)O)=O)cnc2ncnn2c1 C1(CNC(=O)CC2CN3CCC2CC3)CCCC2(CN(C(C3CCOC3)=O)C2)O1 N1(Cc2ccc(C#C)s2)CCC(O)(C(=O)NC2CCC(O)C2)CC1 c1(CNC(=O)C(=O)NC(CNC(c2ccncc2)=O)CO)ccc2nc[nH]c2c1 C(C(=O)NCCOC1CCN(C(c2cnc(C)nc2C)=O)C1)(C(C)(C)C)OC N1(C(c2ccc(C#C)o2)=O)Cc2ccnn2CC(NC(=O)C(CC(C)C)OC)C1 c1(C(=O)NCC2(C)CCCN(C(CCSCCCC)=O)C2)cc2cnn(C)c2s1 c1(OC)ccc(COC(C2(S(C)(=O)=O)CCCC2)=O)c(Cl)n1 CC(CC(=O)N1CCC(OC2CN(C(C34CC(CO)(C3)OC4C)=O)C2)CC1)C(F)F CS(=O)(=O)c1ccc(C(=O)NNc2ncnc3[nH]cnc23)cc1 C1(C(=O)NC(C(C)NC(C(CC)(CC)CO)=O)CO)CCCN2CCCCC12 c1(C(N2CC(NC(C=CC(CC)C)=O)C(C)C2)=O)ccc(C(C)(F)F)nc1C c1(C(=O)NCC(C)N(C)C(C2(C#N)CC=CC2)=O)cc2cc(N)ccc2o1 N1(C(CCOCC)=O)CCC2(NC(=O)CCCC(F)(F)F)CCCC12 c1cc(-c2ccc(C(F)(F)F)cc2)c2nccn2c1 n1(CC=C)cc(C(N2CC(NC(C3CC3c3ccsc3Br)=O)C2)=O)nn1 Cc1cc(C(N2C(C(F)(F)F)CCC2C)=O)nc(Cl)c1.n12c(cccc1=O)CCC2 c1(OC)nc(Cl)c(C(=O)N(C2CN(C(=O)CC3(C)CC3)CC2F)C)s1 C1(NCCNC(=O)NCc2cc3ncn(C)c3cc2)COc2ccc(Cl)cc2O1 c1(OCCCNC(C(=O)NC(C)(C)CN2CCCN=C2N)=O)ccc(F)c(F)c1 C12(CC(=O)NC3CCCC(NC(C(CSC)O)=O)C3)CCC(CC1)OC2 C12(N(C(c3ccc(Br)cc3)C(=O)NC3CCCC3)C)CCC(C#N)(CC1)CC2 c1(C(N2C(CN(C(Cc3ccc(C)s3)=O)C)CCC2)=O)cc(C)cc2ccoc12 C1(NC(CCC(=O)NCC)=O)CC(CNC(=O)CC(=O)NCC2CC2)C12CCC2 c1(CC)cc(N2CC(NC(C3(C4CCCO4)CC3)=O)CC2C)ncn1 C1(CNC(C(C=CC)O)=O)CC2CC(C1)N(C(c1ccc(C#N)cc1C)=O)C2 C(=O)(CCCS(C)(=O)=O)NCC1C2N(C(C3ON=C(C)C3)=O)C(CC2)C1 C1(NC(Cn2c(C)cnc2)=O)CCN(C(c2cnc(C3CC3)[nH]2)=O)CC1C(C)C N1(C(C2(C)C=CCCC2)=O)Cc2ccccc2C(NC(C2CCCCCC2)=O)C1 C1(O)(CNC(CCC(=C)C)=O)COC2CC1C2 c1(C(N2CCC(C(C)NC(C3CCC34CCC4)=O)CC2)=O)ccc(S(C)(=O)=O)[nH]1 c1(C(N2CCN(C(c3ccc(Cl)cc3F)=O)C(CO)C2)=O)ccc(Br)c(Cl)c1F c1(OC)c(O)cc(C(=O)NC2CC(NC(c3cc(C(F)(F)F)no3)=O)C2)cc1O Cc1cc(NNC(=O)Nc2ccc3nc(CN(C)C)[nH]c3c2)nc(CO)n1 CN1CCC2CCN(C(C3CCN(C(C4CCCN4C)=O)CC3)=O)C2C1 c1(CNC(C(=O)OCC)C)c[nH]nc1Br c1(OC)nc(Cl)ccc1CC(=O)NC1CC1NC(C1CCN(CC(C)C)C1)=O N1(C(C(C2(C3(O)CCOC3)CC2)NC(=O)CC(=O)N2CSC2)=O)CCN(C)CC1 c1(N(CCCOCC)C)nc(=NC(C)c2ccc(C)o2)[nH]c2ncn(C)c12 C1(OC)CC(F)CN(C(=O)C(F)C2CC(NC(C3COCOC3)=O)C2)C1 c1(CN2CCCC(C(=O)Nc3cncc(C)n3)C2)c(N)cccc1F C1(CC(=O)NCCOCCC(C)C)CN(C(C2NC(=O)OC2C)=O)CCC1C c1(N2CCC(CN(C(Cn3cc(CC(C)(C)O)nn3)=O)CC)C2)ccc(F)cc1F CC(C)C(F)C(=O)N1CCN(C2CCN(C(=O)Cc3csc(Cl)n3)CC2)CC1 Cc1ccc(CN2CCC(C)(C(=O)NC(c3ccsc3)C)C2)c(F)c1F C(=O)(C(CNC(=O)Cc1ccon1)C(C)(C)C)Nc1c(C)cc(O)nc1 N1(C(c2n(C(C)C)ccc2)=O)CC(CNC(C2CCCC2F)=O)CCC1C CC(C)C(O)C(=O)NCCC(C)(C)CNC(=O)CCC(=O)c1ccc(F)cc1 Cc1nc(=NC(=O)CN2CC(O)CC2c2cccc(Cl)c2Cl)o[nH]1 N1(C(c2nc3sccn3c2Cl)=O)CCC2C(CCCN2C(C2C=CCC2)=O)C1 N1(C(CCC(=C)Cl)=O)CCN(C(C2CCC(C#N)CC2)=O)C(c2ncc[nH]2)C1 c1(NC(CC2OCCN(Cc3c(C)nc(CC)[nH]3)C2)=O)cccc(F)c1C Cc1c(CN2CCN(C(c3ncnn3C)=O)C(C#N)C2)sc2ccccc12 C1(CC)CN2CCN1C(=O)COC(C)C2=O.c1(C(=O)OCCCF)ccoc1C C1(C(N2CC(CC3CC3)C2)=O)(OC)CCN(C(C2CCSCC2)=O)C1 N1(C(C)=O)CCC2CC2(NC(c2cn(C3CC3)nc2C)=O)CC1.C12(CC1)C(=O)O2 c1(C(N2CCCCC(NC(C3(OCC)CCOC3)=O)C2)=O)c(C)nc(=N)[nH]c1C c1(C(=O)NCCN(C(c2cscc2F)=O)CC)ccc(F)c2ccoc12 c1(C(N2CC(OCC(=O)N(CCCC)C(C)CC)C2)=O)ncccn1 N1(C(CC(C)O)=O)CC2CCC1C1CN(C(c3cccnc3N(C)C)=O)CC21 c1(C(=O)NC(C(C)NC(=O)C(=O)NCC(F)F)C)c(Cl)cncc1Cl C1(C(=O)NC2CCCC(O)CC2)CCOCCN1C(=O)C=CC1CCCC1 CCC(C)C1C(=O)NC2(CC2)C(=O)N1C.n1(CCNC(N)=O)ccnc1C C#CCCN=C(NCC(C1(COC)CCCC1)C)NC1CCCC1 c1(OC)ncc(C(N2CC(NC(=O)C3CC3)CC2(C)C)=O)cc1C(=O)O CCCC(C)(C(=O)OCC)NC(C1COC(=O)C1)=O C(=O)(CC(CC)C(F)F)N1CCN(C(c2cnc(CCC)s2)=O)C(CCC)C1 c1(C(N2CC(NC(C=CC(CC)=CC)=O)C2)=O)ccnn1-c1ccncc1 C1(C(N(CCCC)CCCC)=O)CN(C(=O)C(C(C)C)OC)CC12CCC2 C(=O)(CC(C)P(C)(C)=O)N1CC(CCNC(C(CC=C)(F)F)=O)C(C)C1 c1(C(N2CC3(C(NC(CN(C)C(N)=O)=O)CCC3)C2)=O)ccc2c(c1)NCCC2 C(N=c1cc(C)c(C#N)c(C)[nH]1)C1(O)CN(Cc2ccc(OC)nc2)C1 C(=O)(C1=C(Cl)CCC1)N1CCC(CNC(C2(C(=O)OC(C)(C)C)CCCC2)=O)C1 C(=O)(C1=CCN(C(=O)COc2cccnc2)C1)N(c1c(C(C)C)noc1)C(C)C C1(NC(CCNC(=O)OC)=O)C2CC(NC(=O)CC3CCOC3(C)C)CC12 N1(C(=O)NC2C(CC)C3CCC2C3)CC2CC1C1OCCOC21 Cn1nc(Cl)cc1NC(C1CC2CC2N1C(=O)CN1C(=O)CSC1=S)=O c1(C(C)F)ccc(C(=O)NCC2(F)CCN(C(=O)C#CC(=O)N(C)C)C2)cc1 C1(NC(c2c(C)n[nH]c2)=O)CC(NC(C2CC23CCCC3)=O)C(O)C1 c1(C(CNC(=O)CC2(O)CCC2)NC(C2(OCC)CCC2)=O)ccccc1 C123CCCC1N(CC2)C(=O)CN3.C1(CC)CC(CC(=O)N)C1.C(COCCOC)O N1(C(C2=C(C)CC2)=O)CCC(C(=O)N(C2CCCCCC2)C)CC1(C)C c1(CC(N2C(CNC(C=C(CC)C)=O)CC(F)C2)=O)cc(Br)ccc1C C1(C)(CC=C=C)CCN(C(=O)C(=O)NCCNC(c2ccccc2)=O)CC1 n1(CCN(C(=O)CCNS(C)(=O)=O)C)cc(-c2ccc(Cl)s2)nn1 c1(OC)cc(CNCC2CC3CC2C3)ccc1OCC(=O)N(C)C c1(C(=O)NC2C=CCN(C(C3(C#N)CC4(CC4)C3)=O)C2)cnc2ncnn2c1O N1(C(c2cc(C)n(C)n2)=O)CCCC(NC(=O)CCC2CCC(=O)N2)CC1 Cc1ccc2[nH]c(C(=O)NCC(CNC(=O)C=CC(C)(C)C)CO)cc2c1C C1(NC(C)=O)CC2CN(C(=O)C=CCCC(C)C)CCN2C1 C1(CC(C)C)CCCN(Cc2ccc(I)s2)C1 C1(NC(C(C)Cc2ccco2)=O)CN(C(C2(C)CCOCC2)=O)CC1(C)C Cc1nc(CC(C)C(=O)NCCc2cnccn2)oc1C(=O)O.C(C)(C)(C)NC(=O)O Cc1ccc(OCCC(=O)NCC(CNC(=O)C2=CCOC2)OC)cc1 c1(C(=O)NC2CC(CNC(c3ccc(C#C)cc3)=O)C2)cc(C)c(Cl)cc1OC c1(C(=O)N(C2CC3CCC(C2)N3)CC2CCC(F)C2)cccc(Cl)c1F c1(C(=O)NCCCCCNC(c2cncc(N)n2)=O)cc2ccc(Cl)cc2o1 C(=O)(C1=NOC(C)(C)C1)NCCCOCCC(=O)NC1(CC=C)CCCC1 O=C1CCC(CCC(=O)N2CCC3CCCCCC3C2)=NN1.C1CN1 c1(C(=O)NCC2CCN(C(c3ccc(OC)nc3)=O)C2)cc(F)c(C=C)cc1 C1(C(N2CCC(N(CCCC)C(C3CC=CCC3)=O)CC2)=O)COCCC1(F)F CC1CCCC(C(N2CCN(C3CN(C(c4cc(CCO)on4)=O)C3)CC2)=O)C1 N1(C(CCNC(=O)NC)=O)CC(C)(CNC(C2(F)CCCCC2)=O)CC1(C)C Nc1cc2[nH]c(O)nc2cc1C(=O)NCC1CN(C(c2csnn2)=O)CCO1 C=C=C(C)CC(=O)NCC1CC(NC(=O)C(=O)NCCNC(C)=O)CC1O c1(CN2CC(CCF)NCC2)ccc(F)c(F)c1Br Cn1cc(CC(=O)NCC2CC2NC(c2ccc(CO)s2)=O)cn1 c1(CC(N2CCCC(C3N(C(COC)=O)CCC3)C2)=O)c[nH]c2c(F)cccc12 c1(C(=O)NC(C)CN(C(=O)C(F)C2CCOC2)C)ccnn1C(C)(C)C N1(C(CCN(C(Cc2cc(C)nn2C)=O)C)=O)CCc2cc(F)ccc21 CC(CC(=O)N(C1CCC(NC(C2(CF)CC(F)(F)C2)=O)CC1)C)C(F)(F)F c1(C(N2C(C(=O)NC(CC#C)CCOC)CCC2C2CC2)=O)cc2ccccn2c1 C1(NC(c2c(C)n[nH]c2)=O)CC2CCC1N2C(c1cnn(C)c1C)=O O=C(CCCCC(F)(F)F)NCC(C1CC1)NC(C1(C(=O)OC)CC1)=O N1(C(CC(COC)(C)C)=O)CC2(CCN(C(c3nc(C(C)C)no3)C)CC2)C1 N1(C(c2cnc(C(F)F)s2)=O)CCCC(CNC(=O)C(F)(F)c2nccs2)CC1 CC(N=c1[nH]c(=NC(C)C(F)F)c2sccc2[nH]1)c1ccc(C(F)(F)F)cc1 N1(C(CC(CCC)(C)O)=O)CCC2CCN(C(=O)Cc3c(C)noc3C)C2C1 C1(NC(=O)CCc2ccc(F)nc2)CCN(C(C2CC23CCOCC3)=O)CC1O N1(C(c2cc(C)sc2N)=O)CCC(NC(=O)CC(C)c2ccncc2)C(F)C1 C(C(C(=O)NCC(C)(C)n1ccnc1)NC(=O)C=NOC)OCC c1(OC)cc(N2CCCC(C)(C)C2CNC(c2coc(Cl)c2)=O)ccc1[N+](=O)[O-] c1(C(N2C(C)(CC(=O)NCC(C)OCC#C)CC2)=O)ccncc1O C1(C(C)(C)C)CN(C(C2CCC2)=O)CC1(F)CO.c12ccc(cc1)C(=O)NC2 CS(=O)(=O)c1ccc(C(=O)NC2CCSC2)c(Cl)c1.C12(CC1)C(=O)N2 CCC(C)C(O)C(=O)NC1(C(N2CCN(CC)C(=O)C2)=O)CC(O)C1 N1(C(C2C(C#N)C2)=O)CC(NC(=O)CCOc2ccccc2)CC2(CCC2)C1 c1(C(=O)NCCC2CCN(C(CC(C)C)=O)C2)ccc(Cl)c(Br)c1 c1(C(=O)NCC2(NC(CC3(C)CC3)=O)CCOC2)c(S(N)(=O)=O)cnn1C c1(CN(C(CCN(CC=C)C(c2ccn(CC)n2)=O)=O)C)nc(=O)o[nH]1 c1(C(=O)NCC2CC3CC(C2)N(C(=O)CC2CCOC2)C3)n[nH]c2c1CCCC2 C(=O)(C(CNC(=O)CN(C1CCC1)C)OC)N1C(C(=O)OC)CC1 C1(CCOC)CN(C(=O)CC2CCCC2OC)CCN1C(c1ccccc1)=O c1(NC(C(=O)NCCNC(CC)(C)C)=O)cccc2c1CCN(C)CC2 C1(CC(=O)N(C(C)C(=O)NCC(C)CO)C2CC2)CCCC2CC12 C(C(=O)OC(C)(C)C)(C(=O)NCCCC(C)NC(c1ccnc(C)c1)=O)OC n1(CC(N2CC(CCNC(=O)C=Cc3cocn3)(OC)C2)=O)ncc(Cl)c1C C1(C)(C(=O)Nc2cn(CCC#C)nc2)CC(O)CN1C(c1cc(C)c(O)nn1)=O C1(CNC(C2CC(C)OC2)=O)CCN(C(c2ccc(F)cc2)=O)C(C)C1 N1(c2cccc(OCC)n2)CCCC(C)(C(=O)NCc2ccn(C)n2)C1 CC(C)C(CCN(C(=O)Cn1ncnn1)C)NC(C1C(C)C1C)=O Cc1nn(C)cc1C(=O)NC1CN(C(C2CCCCO2)=O)CC1C N=c1nc(Cl)cc(C(=O)NC2CC(CNC(C3CCCCC3C(F)(F)F)=O)C2)[nH]1 c1(C(C(=O)NC(CC)C2CC2)N(C)Cc2cncn2C)ccc(Br)c(Cl)c1 c1(OCCC)ccc(Br)cc1CNCC1CC12CC2.C12CCCCN1C2=O N1(C(CN(C(C(C)C)=O)C)=O)CCC(NC(=O)CC2CCNC(=O)C2)C(O)C1 C1(C(=O)NCCc2c(C)noc2C)C(C2CC2)CCN1C(c1sccc1F)=O C#CC1(C(N2CCC(CCF)CC2)=O)CCN(C(c2ccccc2NC)=O)C1 N1(C(Cn2ncc(C(=O)OC)c2)=O)CCC(NC(c2cc(C)no2)=O)C1C c1(NC(CC#C)=O)n[nH]c2c1CN(C(c1nccnc1Cl)=O)C2 C12(CC(N3CCCC3CNC(=O)Cc3cncnc3O)=O)CCC(CC1)C2 C1(SC)CCN(C(C2CCOCC2NC(C2(C)CCCO2)=O)=O)CC1 C(CCCCCNC(c1ccnn1CC)=O)NC(C(=O)NCC)=O C=CC(C)(CC)C(=O)NCCCN(CCCNC(=O)CN(C)C(C)=O)C C1(N(C(C2CC2F)=O)CC)CCCN(C(C2COCOC2)=O)C1 C(C1=NOC2CCCCC12)N1CCOCC(C(N(C(c2ccccc2)C)C)=O)C1 C1(CC(=O)NCCC(C)NC(C2CCCOC2C2CC2)=O)CCN(CCF)CC1 C1(NC(c2cc(SC)oc2)=O)CC2CC1N(C(c1ccn(C)n1)=O)C2 C(=O)(C1=CCCCO1)NCC1N(C(c2cc(CC)c(C)s2)=O)CC(O)C1 C12(NC(C=CC(C)(C)C)=O)CCCC1CN(C(=O)CC1(C(F)(F)F)CNC(=O)C1)C2 C1(C(N2CC(CC(=O)N(CC#C)CC)OCC2)=O)CCC2(CCC2)C1 c1(C(N2C(C)CC(NC(c3cc(CN(C)C)on3)=O)C2)=O)cc(O)ccc1N N1(C(CN(CCOC)CC)=O)CCOC(C)(CNC(C2CCC(F)(F)CC2)=O)C1 N1(C(c2cccc(NC)n2)=O)CC2CCC1C(NC(C1CN(C)CC(C)O1)=O)C2 C(=O)(C(C)C(F)(F)F)N1C(C)CC1C(=O)NCC1CCCOCC1 c1(CCC(=O)N(CCCC(=O)O)CC)ccc(-c2cc[nH]n2)cc1 CCCCC(F)C(=O)NC(C1CCN(C(=O)Cn2nc(C)oc2=O)C1)C(=O)NC CC1(CNC(C2COCCO2)=O)CCN(C(=O)CNC(=O)CCCCO)CC1 C(c1ccn(C)c1)=CC(=O)N(CCNC(CCCN(C(C)=O)C)=O)CCN(C)C N1(C(CNC(CNC(CC=C=C)=O)=O)=O)CC2(CC(OCC(C)(C)OC)C2)C1 c1(C(N2CCCC(CNC(C3=CC(C)CC3)=O)C2)=O)ccc2cc(Cl)ccc2c1 c1(N2CC3CN(Cc4cccc(OC(C)C)c4F)C3C2)ncc([N+](=O)[O-])cc1Br c1(OC)cc(N2CCC(N(C(=O)C(C)C3CCOC3)C)CC2)ccc1[N+](=O)[O-] c1(NCC(CNC(C2(C(=O)NC)CC2)=O)O)cnc(F)cn1 N1(C(CCc2ccc(OCC)nc2)=O)CCCC(C)(CN=c2[nH]ncs2)C1 c1(C(C(=O)N(C)CCOCCNC(=O)C(O)c2cnc[nH]2)(C)C)cncc(F)c1 C1(CC(=O)N(C2CN(C3CC3)C2)C)CCCN(C(=O)Cn2cccnc2=O)C1 C(CNC(C1(F)CC1)=O)(CC(F)(F)F)NC(c1cn(C)nc1C(F)F)=O c1(OC)cc(C(N2CC(NC(C3C=CCC3)=O)C(C)C2)=O)ccn1 C1(NC(C(c2scc(C)n2)C)=O)CCN(C(C23CCCC2(C(N)=O)C3)=O)CC1 C(C)(C(CC(=O)NC(C1CSC1)C)NC(C1CC(C(N)=O)C1)=O)OC c1(C(N(C)CC2N(C(c3cc(C)ns3)=O)CCCC2)=O)csc2cncn12 C(c1c(NC(=O)C(C)C)nc2ccccn12)=CCNc1c(C(=O)OC)cccc1 c1(C(N2CCCC(N(C(c3nnn(CC)c3C)=O)CC)C2)=O)c(F)ccc(F)c1O C1(CC#C)CCN(C(C2(CNC(C3CCC(=O)O3)=O)CCCO2)=O)C1 c1(OC)cc(C(=O)NCC(CCNC(c2csc(C)n2)=O)OC)ccc1F CC(Cc1ccccn1)(C(=O)O)NC(=O)CCSCC(F)C(F)(F)F N1(C(C(CC=C)C)=O)CCC(NC(=O)C=CS(=O)(=O)CC)C2(CCC2)C1 C(=O)(C1=CCN(C(C2C=CCN2)=O)C1)Nc1c(C(=O)OC)cnn1C c1(N(C2CC23CCNCC3)C(C2CCCC(C)C2)=O)ncc2cn[nH]c2n1 CC1CC(C(=O)N(CCNC(C23CSC(C2)C3)=O)C2CC2)c2ccccc2N1 c12cnc(nc1)N1CCOCC1CC(=O)N2.c1(CC)csc(C(=O)OC)n1 c1(NC(=O)NC(CC)C(=O)NCCOCCN(C)C)c(Br)cccc1C CCCC(C(=O)N1CCOC(C(=O)N(C2(C)CC2)CCC(C)C)C1)S(N)(=O)=O N1(C(C2C(CC)OCC2)=O)CC2(CCN(C(=O)C(C)(C)COCC(F)F)CC2)C1 c1(C(=O)NCC(N2CCC2CNC(C2CC(O)C2)=O)=O)cc(F)ccc1F C1(CC(=O)NCCN2CCCCC2=O)CC2(CC2)CN1C(=O)CC1CCCOC1 C(C)(CCCC(=O)NCc1ncn(C2CC2)n1)NC(C1N(CC)CCCC1)=O C(=O)(C(C)(CC)CC)NC(CCC)CNC(=O)C(c1cccnc1)O C(=O)(C1CCCc2cccnc21)NCC(CCOC)NC(C(CC)OCC)=O C1(C(=O)NCC(=C2CN(C(C3(COC)CC=CCC3)=O)C2)F)CCOC(C)(C)C1 c1(C(=O)NCCCN(C(CC=CC)=O)C2CC2)nn(C)c(C2CC2)c1C N1(C(CCc2c(C)noc2C)=O)CCC2(CCC2NC(=O)CC#N)CC1 C1(CC(C)=O)(C(=O)OC(C)(C)C)CCCN(C(=O)C(C)CN(C)C)C1.C(=O)(N)OO.O C1(CC(C)NC(C(C(C)C)OCC)=O)CC2CCC(C1)N2C(c1cccn1C)=O Cc1ccc2c(=NC3CC(F)(F)C3)[nH]c(=NCC3CCC(C)(C)C3)[nH]c2c1 c1(OC)ccccc1NC(=O)C(C)NCC1(c2nc(C)cs2)CC1 c1(C(=O)NC2(C)CN(C(c3scc(C)c3C)=O)C2)cc2cnccc2cc1F N1(C(c2c(C)n(C3CC3)cc2)=O)CCC2(CO)CN(C(C3(F)CCC3)=O)CC2C1 c1(C(N(C2CCCN(C(C3(Cl)CC3)=O)C2)CC)=O)cccc(C(C)(C)C)c1 CCC(O)C(F)(F)C(=O)NCC1CC2CCC(C1)N2C(=O)CC1CCS(=O)(=O)C1 N1(CCC(=O)NC2CN(C(=O)CNc3nccs3)CC2O)CCCCC1=O CCS(=O)CC(=O)NCC(C(F)(F)F)N1CCN(C(=O)Cc2ncoc2C)CC1 C1(NC(=O)C2=COCCO2)CC2CC1CN(C(c1cnccc1Br)=O)C2 N1(C(COCc2cc(C)on2)=O)CCOCC1CCNC(C1CNC(=O)N1)=O C1(C)(C(N(C)CC2N(C(c3c(C)nc[nH]3)=O)CCCC2)=O)CCCC(F)(F)C1 c1(NC(C(c2cccc(Cl)c2)C)=O)cc(-c2ccccc2)sc1C(=O)O CCCC(C)(C)C(=O)NCC(C)CNC(=O)C(O)CCSC Cc1cc(O)cc(=O)n1CCC(=O)N(C1CCCN(C(C2CC(C)(F)C2)=O)C1)C N1(C(c2c(CC)nn[nH]2)=O)CCN(C(=O)CSC)C(C)C1 C1(C(=O)NCC2CCC(=O)NC2C2CCCC2)CC2CNCC1C2 N1(C(C(C)(O)C2CC2)=O)CC2CCN(C(=O)C3=NN(C4CC4)C(=O)CC3)CC2C1 C1(C(=O)NCCCC(C)(C)F)CC2(CC(NC(C3NC(=O)OC3C)=O)C2)C1 CCCC(C(=O)NC1CC(NC(=O)C2=CCC2)C1)c1ccc(Cl)cc1 c1(N2CCCCC2=O)ccc(Br)cc1F.N1(CC(C)CNCC(=O)NC)CCCCC1 C#CC(C)(C)C(=O)NC(CNC(c1cccc(C2(C#N)CC2)c1)=O)C(C)(C)C c1(OC(COc2c(OCC(C)C#N)cccc2)=O)ccc(Br)cc1Cl C1(CC(=O)Nc2cccc(C(F)F)c2)CC(O)CN1C(c1ccc(CO)s1)=O C1(=O)CC(O)CCSC2(CCC2)C(=O)N(C2CC2)CCN1.c1(CC)ccccc1.COC CC(C)C(C(=O)N1CC(C)(N(C)C)C1)C(C)NC(=O)COc1ccsn1 C1(C(=O)NCC(=C)CCNC(=O)CCNS(=O)(=O)C(F)(F)F)CCC(C)NC1=O C1(NC(C(CC)NC)=O)CC2(CCN(Cc3ccccc3C(F)(F)F)CC2)C1 C(CC(=O)N1CCC1)N(C1CCSC1)C(C1C=CCC1)=O C(=O)(CC(C1=CCCC1)OC)Nc1cncc(OCC(=O)NC)n1.OCC C1(C(N2CCN(C(C)=O)CC2)=O)CC(N=[N+]=[N-])CN1C(=O)C(N1CCOC1=O)C c1(CC)ccccc1C(N1CCC(C(C)(O)CNC(=O)CCOC)CC1)=O C=C(C)CC(C)C(=O)NC1CN(C(=O)Cc2cc(F)ccc2OC)C(C)(C)C1 c1(C2C(C(=O)NCC(CC)NC(CC=CCC)=O)C2)cc(F)cc(Br)c1 N1(C(c2ccc(C(C)C)o2)=O)CC(NC(=O)C(C)S(N)(=O)=O)CCC1C c1(C(N2CCC(C(C)NC(c3c(CC)nns3)=O)C2)=O)cnc2cnn(C)c2c1 N1(CC(=O)NC2C=CC(C(=O)NCc3ccc(C)nc3)C2)CCS(=O)(=O)CC1 C1(CNC(C2C=CCCC2)=O)CCCN1C(=O)C=Cc1ccco1 c1(C(N(C(CNC(CC(C(=O)OC)C)=O)C)C)=O)cc2c(s1)CN(C)CC2 C(=O)(CCCC(F)(F)F)NCCCC1N(C(=O)C2=CSCS2)CCCC1 c1(-c2cn(C(C(C)O)C)nn2)cnn2c1CN(C(c1c[nH]nc1C1CC1)=O)CC2 c1(C(N2CC3C(CNC(C4(SC)CCC4)=O)C3C2)=O)cnc2ccoc2c1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CCN(C)C(C(=O)NC2C=CCC2)C1 N1(C(=O)Nc2cc(SC)ncn2)CCC2(CCC(OC)C2)C1 N1(C(c2c(C)sc(O)n2)=O)CCC2(C1)CN(C(=O)C(C(C)C)NC(C)C)CCO2 c1(OC)c(OC)ccc(COC(=O)C(F)(F)c2csc(C(F)(F)F)n2)c1[N+](=O)[O-] CC1(C)CCCC1C1CCN(CC2CC3CCC2C3)C1 C(C(C)(C(=O)NC(C1(CNC(c2nc(C)oc2C)=O)CC1)C)OC)OC.C(C)(=O)N c1(CO)ncccc1F.c12ccc(cn1)C1C(C1)C(=O)N1CCCC1CO2 C(=O)(C#CC1CCCOC1)N1CC(CC)N(C(c2nnn(CC)c2C)=O)CC1 c1(OCC)ccccc1CCC(N1CC(NC(c2cnn(C)n2)=O)C(O)C1)=O CC(C)(C#N)CCC(=O)N1CCN(C(=O)C=Cc2cccs2)C(c2cn[nH]c2)C1 CN1CC2(CC2)CC1C(=O)NCC1CCN(C(c2cc3[nH]ccc3s2)=O)C1 S(=O)(=O)(c1cccnc1NCCOC1CC1)NC1C(C)N(C)CC1 c1(CNC(c2cccc(OCC(C)C)c2)C)ccc(S(=O)(=O)C2CC2)cc1 c1(C(=O)NCCCC(C)NC(c2cccc(C#N)c2)=O)c2c(nn1C)CCOC2 Cc1nc(S(=O)(=O)NCCC(=O)NCCC(C)(C)NC(C2CCSC2)=O)cn1C C(=O)(CC(C)(C)C)N(C)CCOCC(=O)NC(C(C)(C)O)C1CC1 c1(C(=O)OC)ccccc1NC(C1CCC1NC(c1cnnc(Cl)c1)=O)=O c1(CC)ccc(C(=O)NC(C)(CC(N2CCCCC2C2(O)CC2)=O)C(C)C)nc1 c1(OC)nc(C)ccc1C(N1CC=CCC1n1cc(C(=O)N(C)C)nn1)=O C(CCCC(=O)NC1CC1(c1ccco1)C)N(C(C)(C)C)CCO C1(NC(c2c(C(C)C)occ2)=O)CC2CCC(C1)N2c1nc(Cl)ncc1Br Cc1cc(OC2CCC(OCc3ccccc3)CN2)nc(C)c1 N1(C(CNC(=O)NC)=O)CCC(F)(CNC(=O)COCc2ncnn2C)CC1 c1(NC(C(N)c2nccs2)=O)cccc2c1C(=O)NC2=O CC(c1cccs1)=CC(N1CCN(C(=O)CCC(=O)c2cccnc2)CC1)=O CCC(CC(=O)NC1CCC(CC(=O)NC2CCSC(C)C2)CC1)C1CC1 N1(C(CC2N(CC)C(=O)CC2)=O)CCN(C(c2cccc[n+]2[O-])=O)C(CF)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CCC(NC(c2c[nH]c(=O)cn2)=O)CC1C C#CCCCC(=O)NCC1(F)CN(C(=O)CCOCCOC)C1 C1(C2N(C(=O)N(c3ncccn3)C3CC3)CCC2)CCN(C(=O)C(F)(F)Cl)CC1 N1(C(N2C(C)CC(NC(=O)OC(C)(C)C)C2)=O)CCOc2ccccc2C1 N1(C(=O)CC2CCN(CC3CC3)C2)CC2CC1CC21OCCO1 C1(C(N2C(CNC(CCC(=C)C)=O)CC3CC32)=O)CCc2ccccc2CC1 CC1(C)C2CCC(C2)C1NC(=O)CCCCNC(C1CC12CC2)=O C1(CCC(=O)N(CCN=[N+]=[N-])CC)CCN(C(=O)CN2CCCC2=O)C1 C#CCC(C)(C(=O)NCCN1CCC(CO)C1)NC(=O)CC1CCC1 C1(C(=O)NCC2(O)CC(NC(c3cnsc3)=O)C2)CCC2CC2CC1 C1(C(=O)NCCCC(C)(C)C)N(C(c2cccnc2O)=O)CCCC1(C)C N1(C(C2(C)C(C)OCC2)=O)CCC=C(CNC(C2(C)CC2C)=O)C1 c1(OC)cc(NC(C2(CO)CCN(C(=O)Cc3ccccc3F)C2)=O)ccc1C N1(C(=O)Oc2ccc(CC)cc2)CCCc2cc(OCCN(C)C)ccc21 Cc1ccc(NC(=O)C(=O)NC(c2cnn(CCOCCO)c2)C)n1C CN1CCN(C(C2(CF)CCN(C(=O)Cn3cc(C#N)cn3)C2)=O)CC1C1CC1 C1(COC)CN(C(=O)CNC(N)=O)CCN1C(=O)CN1CC2CC2C1 N1(C(CNC(CCCOCC)=O)=O)CCOC(C2(C)N=N2)C1 c1(C(=O)NCCC2CCN(Cc3n(C)ccn3)C2)ccc(Br)cc1CC(=O)O C1(C)(C(=O)NC(C)(C)CCNC(c2scnc2-c2ccccc2)=O)CCNC1=O CC1CN(C(=O)CCc2cnn(C)n2)CC(C)N(C(c2[nH]ccc2C2CC2)=O)C1 Cn1c(O)nc2cc(C(=O)NC3(C4CCCN4C(C4CC45CC5)=O)CC3)cnc12 C1(CC(=O)N(C)CCc2cc[nH]n2)CC(NC(c2cc(O)ncn2)=O)C1(C)C N1(CC(N2CCC(CNC(CCC3CCCN(C)C3)=O)C2)=O)CCCNS1(=O)=O C(=O)(C1=CCC(C)CC1)NC1C(CNC(CCc2ncc(C)[nH]2)=O)CC1 c1(CN=c2ccnc(N(C)CCC3CCCC3)[nH]2)cc2ccnc(F)c2o1 Cc1nnc(O)c(C(=O)NCC2(C)CCN(C(C3CCOC(C)C3)=O)CC2)c1C N1(C(c2c(CC)nc[nH]2)=O)CC(OC)CC1(C)CNC(c1nnn2c1CCC2)=O CN(CCCC(=O)N1CCN(C(C23CC(N=[N+]=[N-])C2C3)=O)CC1C1CCC1)N=O N1(C(c2cc(F)c[nH]2)=O)CCCC2(CCCN2C(c2cc(F)cc(Br)c2Cl)=O)C1 CC(CC(N)=O)C(=O)N1CCC(NC(=O)COCc2ccnc(O)c2)C(C)C1 n1(CC)ccc(C(=O)NCC2(F)CC(CNC(C3(C)CC=CC3)=O)C2)cc1=O C1(NC(=O)CCn2ccnn2)CC(CNC(C2(C(=O)NC)CCC2)=O)CC1O c1(CNC2CCCN(C(=O)NC3(C#N)CC(N(C)C)C3)C2)nc(Cl)ccc1Cl C#CC1CN(C(c2cncn(C)c2=O)=O)CCN1C(=O)CNC(=O)CC(C)C C1(C(N2C(C(N(OC)C)=O)CSC2)=O)COC(C)(C)OC1 O=C1C=C2CN(C(C3CC=CCN3C(C3C4CCCC34)=O)=O)CCN12 C(=O)(N=c1[nH]nc(CSc2ccccc2)s1)NC(Cc1cccc(C)n1)C c1(C(N(C(C)C(=O)NC2CCCCC2)CC)=O)cnc(O)c(C)c1 c1(NC(C2(F)CN(S(CCOCC)(=O)=O)C2)=O)cc(OC)cc(Br)c1 C=CCC(CC(=O)OC)NC(=O)C(F)(F)CCn1cc(CCNS(N)(=O)=O)nn1 C(C(CC1CC1)CO)N1C(=O)C2(CC2)C1.c1(NC(=O)CCN2CCC2)ccccc1 CC1(C)CC2(CC2C(=O)NC2COCCN(C(c3cnn(CCF)c3)=O)C2)C1 N1(Cc2c(OC)nsc2)CCCC(C(=O)N(C)C(c2cccnc2)C)C1 CC(CC(N)=O)C(=O)NCC1CC(F)(F)CN1C(c1cnn(CC(F)(F)F)n1)=O c1(C2N(C(C)(C)C)CCOC2)nc(N=c2ccn(CC3CCOCC3)[nH]2)cs1 c1(COC(C2CC(CC)OCC2)=O)cnc2cc(OC)ccn12 N1(CCOC)CCC(N=c2[nH]c(=NCCCCOC)[nH]c3cc[nH]c23)C1 c1(SCC)cc(C(=O)NCCC(O)CNC(=O)CCc2nccn2C)ccn1 C12(CC(=O)NCC#CCNC(C3C(C)OCCC3)=O)CCC(CC1)OC2 N1(C(Cc2c(C)nc(C)s2)=O)CCC(C)C(NC(c2cnc(N(C)C)nc2)=O)C1 CC#CC1CN(C(=O)CCCN(C)C(C2CC(CC)=NO2)=O)C1 C(C(F)(F)CCC(=O)NC1CCC(=O)NC1)n1cc(-c2c(OC)cccc2C)nn1 CC(C)C(C(=O)NC1CC(CO)(CO)C1)NC(c1nccn1C)=O C(CC(=O)N1CCC(C(=O)N(C(C)C(=O)NC)C)O1)OCCCOC Cc1cc(Br)c(C(C(=O)NCCCF)N(CC#N)CC2CC2)s1 N1(C(C2CC(NC(c3c(C)cnn3C)=O)C2)=O)CC(C)OC2(CCC2)C1 C=CCC(C(=O)N1CC=CC(NC(=O)CCCCOC)C1)N(C)C N1(C(c2c(O)cc(F)cc2F)=O)CCC2(CCN(C(C3CCOC3)=O)C2)C1 C1(NC(CCSCC)=O)CCCC(NC(=O)CCN(C)CCO)C1 N1(C(CC2(C(=O)OC)CC2)=O)CCC(C)C(NC(C2CCN(C)C(=O)C2)=O)C1 N1(C(C2CCC(C)(C)C2)=O)CCC2CC1CN(C(c1cnc(OCF)cn1)=O)C2 C(CCNC(=O)C=CC(F)(F)F)(C(=O)NC(C(N)=O)C(C)C)OC N1(C(c2[nH]cc(C)c2)=O)CCCC2(NC(C3CC34CCOC4)=O)CCCC12 C1(NC(C(C2CCOCC2)C)=O)CCN(C(=O)COc2cnc(Cl)cn2)C12CC2 CCC(Cc1cnc[nH]1)C(=O)NCC(C1CCCC1)NC(C1(O)CCCC1)=O N1(C(C(CC)SC)=O)CCC2(CCN(C(C3(c4cccs4)CC3C)=O)CC2)C1 C=CC1(COC(C2CC2(c2ccc(C(=O)OC)cc2)F)=O)CCOCC1 N1(C(C(=O)NC(C)C)=O)CCC(NC(c2cccc(C(F)(F)F)c2)C(F)F)CC1 CCC(CC(C)C)C(=O)N1CC=CC1C.C(=O)C(C)(C)CF.c12ccc(cc1)s2 c1(C(=O)NC(CNC(c2cccc3c2CCC3)=O)C2CC2)cc2ccsc2s1 c1(C(C)OC)nc(C(=O)NCCOC2CCN(C(c3scnc3C)=O)C2)cs1 Cc1ccc(Cl)cc1NNC(=O)C(COC(C)(C)C)NC1CCN1C(N)=O CC1CCC(C)(C(=O)NCCCC(C)(C)NC(c2cncc(C(F)F)c2)=O)CC1 C(=O)(C(C(=O)NC1CCC(CNC(=O)C(F)OC(F)(F)F)CC1)OC)OCC c1(OCC(C)C)ccncc1NC1CCCN(c2ccncn2)C1 C(=O)(C1COc2cc(F)ccc21)NCC1(C)CCC(C(=O)O)CC1 CC1CN(C(c2cc(C(C)(C)C)on2)=O)CC(C)C1NC(C1CC2C=CC1C2)=O c1(CCC)cccc(C(=O)N(CC)CC2CCCN2C(c2snnc2C2CC2)=O)c1 CP(C)(=O)CN1CC(C(=O)NCC(F)CNC(=O)CC2CC3(CC3)C2)C1 CCC(CC)(C(=O)N1CC(CCNC(C2CC(F)(F)CS2)=O)C1)C(C)C c1(CC(=O)N(CCNC(=O)C(C)c2cccs2)CC)c(F)cc(Br)cc1F N1(C(C(F)=CC)=O)CCN(C(c2cc(C)cc(Cl)n2)=O)C(CCO)C1 N1(C(C(c2ccccc2)C)=O)CCOC(C(=O)NCCNC(C23CCC(C2)C3)=O)C1 C1(C(N2CCC(OCC=C)CC2)=O)CN(C(=O)Cc2ccnn2C)CC1C1CC1 c1(C(CNC(=O)CC(N)Cc2cccc(F)c2)N(C)C)cccc(C#N)c1 N1(C(Cn2c(C(=O)OC)cnc2)=O)CCC(N(C)C(c2sncc2C)=O)C(C)C1 C1(C(N2C(C(=O)Nc3cncc(CN(C)C)c3)CC2)=O)CCOC2CCCCC12 C1(NC(c2c(NC(=O)CC3CCCO3)ccs2)=O)CCC(C(F)F)CC1 C#CCC(C)(C(=O)N1CC2(CCCO2)C1)NC(=O)C(C)n1ccnn1 C(=O)(C1Cc2ccc(F)cc21)N1CCC2(C(NC(COCC(=C)C)=O)C2)CC1 CC1C(C(=O)N(C)Cc2ncnn2C)CCN1C(=O)CCOC1COC1 N1(C(C2C(CCOC)C2)=O)CC(O)(CCNC(c2conc2C2CCCO2)=O)C1 N1(C(C(C)(Cl)Cl)=O)CCC(CCN2CCN(C(=O)COc3ccsc3)CC2)CC1 C1(NC(CCOC)=O)CC2CC(C1)N(CCO)C2 Cc1[nH]c2ccccc2c1CC(N1CCC(NC(C2CCC(=O)N2)=O)C(F)C1)=O C(C1OCc2ccccc21)NC(c1cccn1Cc1ccncc1)=O C1(NC(COCCOCC#C)=O)CCCC(NC(=O)C(C)=C(C)C)C1 CCN=C(NCCCCCC(=O)OC)N1CCC2(CC1)CC2(F)F CC1OC2(C(N3CCC(C(=O)NC(Cc4ccc(O)cc4)CO)CC3)=O)CC1C2 c1(OC)cc(C(=O)NCCNC(=O)C=CCN2CCCC2)cc(OC)n1 C12(C(=O)NCC(CC)NC(C(CC)N(CC)CC)=O)CC3CC(CC(C3)C1)C2 C=CCCCCCCC(=O)N1CCN(C(c2cnn3ccsc23)=O)C(CCO)C1 C=CCC(C)(C)C(=O)NC1CC(CNC(c2nnsc2C)=O)C1(C)C C1(O)(NC(=O)COC(F)F)CCN(C(=O)CNC(=O)Nc2cccc(O)c2)C1 N1(C(C(c2cccc(C)c2)=O)=O)C2CCC1CC(O)(CNC(=O)CS(C)(=O)=O)C2 c1(OC)cc(C(=O)NC2CN(Cc3ccnc(Br)c3)C2)c(CO)cn1 C1(C(=O)NC2CC(N(C(=O)Cn3ccnn3)C)C2)CCC2(CCC2)OC1 c1(CC(=O)NC2CCC(CNC(CCCOC(C)C)=O)C2)ccc(F)cn1 N1(C(c2scc(COC)c2)=O)CC(C)(C)CC1CNC(C1CCCC(F)(F)C1)=O c1(OC)ccc2c(c1)CN(C(c1cn(C)cn1)C(=O)NC1CC1)CC2 c1(C(=O)NCCC(=C)CNC(=O)CC2(C)CC2)cc(C)c(CC)[nH]1 c1(C(N2CCN(C(C(C)C)=O)C(CF)C2)=O)sc2ncccc2c1Cl Cc1cc(N2CCCC(NC(C3C(C)(C)C3(C)C)=O)C2)nc(C)c1C#N c1(CNC(c2cc(C)oc2C)=O)cc(O)nc(CNC(=O)C(C)OCC(C)C)n1 c1(C(=O)OC)cc(F)c(C(=O)NC(CNC(C2CC2C)=O)C(F)(F)F)cc1F O=C(C1OCCc2cc(Br)ccc21)OCc1nnc(-c2cccs2)o1 c1(CC)[nH]nc(Cl)c1C(N1CC(CNC(=O)C(C)(F)CC)C(O)C1)=O n1(CC)cc(CC(=O)N(CCCNC(C2(Br)CC2)=O)C2CC2)c(C)n1 c1(C(=O)NC2CCC(NC(C(COC)OC)=O)CC2)cc(S(N)(=O)=O)c[nH]1 Cc1cccc(CNC(=O)COC2CCN(C(=O)CCCC#N)C2)c1C C#CCCCCC(=O)N1CCCC(C)(CNC(=O)CCC(F)(F)F)C1 N1(C(=O)CN2CCn3nccc32)CCC(C2(NC(C3(CF)CCC3)=O)CC2)C1 C(=O)(C#CC(C)(C)CNC(=O)C(c1cncn1C)O)NC(CCOC)C c1(C(=O)NCC2CC(c3ccccc3)CO2)cccc2cc(Br)cnc12 CCC(C)C(C(F)(F)F)NC(N1CCC(NC(c2ccc(C)cc2)=O)CC1)=O N1(C(CCCCC=C)=O)CC2(C(=O)NCc3ccc(C)c(Cl)c3)CCC1CC2 C1(OCC)CC2(C1)CC2NC(=O)CC1CC1NC(=O)CCSC CC1CC(CNC(=O)C(CC2CC2)NC(c2nccn2C)=O)CCO1 C(=O)(C(CC(F)F)N(C(=O)C(CO)NC(N)=O)C)NCC1(C(=O)OC)CCC1 CC1(CNC(=O)C=Cc2ccccc2F)CC(F)(F)CN1C(C1CCCCS1)=O C(=O)(C(F)(F)CC1CC1)N(CCCN(C)C(c1ccc(N)cn1)=O)C C(CC1CNc2ccccc21)N(C(C(C(C)C1CCOCC1)N)=O)Cc1ccccc1 c1(C(=O)OC)cc(C(=O)NC(C)CNC(=O)C(C(C)C)N(C)C)c(C)s1 C1(CC(N2CCC(NC(C3C4CN(C)CC43)=O)C2)=O)CC(C)(C)OC1=O CC1(C(N2CCCC(CC(N3CCC(C(C)(C)C)C3)=O)CC2)=O)CC2(CCC2)C1 C(=O)(C1=CC2CCC(C1)C2)NC1(CNC(c2ncc(C)nc2)=O)CCCCC1 c1(C(N2CC(NC(C(CC)CC)=O)C(F)(F)C2)=O)cc(Br)c2ccccc2n1 N(C(=NCCC(C)(C)S(C)(=O)=O)NCc1ccnn1C)Cc1cc(C)ns1 C(=O)(CC(C)C(=O)OC)N1CC(CCC=C)(CCC=C)C1.c12ccncc1C(=O)N2 C(=O)(C(C)(C)CC1CCOCC1)NC1(C2N(C(C3C(C=C)C3)=O)CCC2)CC1 C12(N(C(C(F)(F)F)C3CCCCC3)C)CCC(c3nc(C(C)(C)C)no3)(C1)OC2 C12(C(N3CC(C)(NC(c4cc5oc(Br)cc5s4)=O)C3)=O)CC1Cc1c[nH]nc12 N1(C(C2C(C(C)(C)O)C2)=O)CCC2(CC1)CCN(C(c1sccc1Cl)=O)C2 c1(C(N2CC3C(C(=O)NC(CC)C(N)=O)C3C2)=O)cc(CNC)ccn1 CC1CN(C(=O)OC(C)(C)C)CCC1NC(=O)C(CO)CO c1(CNC(C(C)=C(CC)C)=O)cccc(NC(=O)C(C)n2cccn2)c1 C1(C(N2CC(N(C(=O)C(CO)c3ccccc3)C)C2)=O)CCCCCC(=O)C1 c1(CC)oc2ccccc2c1C(=O)NCC1CC(C)N(C(=O)CN(C)C(N)=O)C1 Cc1nn(C2CCOCC2)cc1NC(C)CCN(C(=O)C=CC(C)C)C CC1(C)C2CCC1(C(=O)NC1CCC(CNC(=O)C(Cl)=CCl)CC1)CC2 N1(C(CC(C)n2cccc2)=O)CC2CN(C(C3(C)CC3(C)C)=O)CC2C1 N1(C(CCC#C)=O)CCC(C)(C(N2CCCC(C(=O)OCC)C2)=O)C1 c1(C(=O)NCCCN(C(c2c(CCC)n[nH]c2)=O)C)sc([N+](=O)[O-])cc1Cl N1(C(C(C)(C)N2CCCCC2)=O)CCC2CCN(C(=O)C(O)CC3CC3)C2C1 CCCC(CC)C(=O)NCC1(C(=O)NCCCC2CCOC2)CC1 N1(C(C)=O)CCCC1C(=O)NC(C)CC(C)NC(=O)C(C1CCCO1)C1CC1 C1(CNC(c2c(C)n[nH]c2)=O)CCN(C(=O)CCC(C)(C)N(C)C)C1(C)C C1(CNC(C2C(C(N)=O)C2)=O)CCN(C(=O)Cc2coc(C(F)F)n2)CC1(F)F CC1(C)C2CCC1(C(=O)NCC(F)(F)CCn1cc(C(C)(C)C(=O)O)nn1)CC2 CCCC(C)(C)CC(=O)NC1CC1NC(c1cc(C2CCCCC2)ccc1O)=O C1(C(N2C(CN(C)C(c3cnn(C)c3Cl)=O)CCC2)=O)CCC(F)(F)C1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCN(CCCNC(C2C(C=C)C2)=O)CC1 C1(NC(COC)=O)CCCN(C(=O)C(O)CC2CCCCC2)C1 c1(-c2c(C)cc(NCc3c(CCOC)cccc3)nc2)cc(F)c(F)cc1O N1(C(C2CCN(CC)C2)=O)CCCN(C(=O)CNC(=O)OC)CC1C C(=O)(C(O)C1=CCCCC1)NC(CNC(c1[nH]cc(CC)c1)=O)CC(F)(F)F C(=O)(C1=COCCC1)N(N1CCC(n2nccn2)CC1)C N1(CC)CCOCC1CC(N1CCC(NC(=O)CCc2ccccc2O)C1C)=O CC(CC(=O)NC1(C)CN(C(=O)C(C)NC(C2CCCC2)=O)C1)C1CCCO1 c1(C(=O)OCC)c(NC(C2(C(=O)NC(=O)C(C)CC3CC3)CC2)=O)csc1C N1(C(CNS(NC)(=O)=O)=O)CC(CO)C2(C1)CN(C(C1CCC=CCC1)=O)C2 C12(CNC(C(C)C(C)(C)C)=O)CCCC(CN(C(=O)C3=CCCC3)C1)C2 N1(C(C(CC)C)=O)CC2CCCC(N(C(=O)Cc3c(C)ncnc3C)C)C2C1 C(=O)(C(C)(C)CNC(=O)CCc1conc1C)N(CC(C(C)C)OC)C CC1(C)CCc2[nH]c(C(=O)NC3CC(O)CN(C(=O)CCC(N)=O)C3)cc2C1 C1(N(C(c2n(C(C)C)ncn2)=O)C)CCC(NC(=O)C(c2ccccn2)O)CC1 C(C1CN(C(c2cc(C(=O)OC)no2)=O)Cc2ccccc21)NC(C(C=C)(F)F)=O C=CCCCC(C(=O)N1CC(C)(OCC(=O)NC)C1)NC(=O)CC1CCOC1 C1(O)(CCNC(c2c(C(C)(C)C)c[nH]c2)=O)CCN(C(c2ccc(O)nn2)=O)C1 C1(C)(C(C)NC(C2C(F)(F)C23CC3)=O)CN(C(=O)CNC(=O)C2CC2)CCO1 c1(NC(C)=O)ccc(C(N2CCC(NC(c3ccc(F)cn3)=O)C2C)=O)nc1 C1(C(=O)Nc2c(C(=O)NC)cccc2)CCC(C)CN1C(C(C)C(F)(F)F)=O C(=O)(CC(C)(C)C#N)NC1(C)CN(C(Cc2scc(CC)n2)=O)C1 C1(SC)CN(C(=O)CCCc2ccsc2)CC1NC(C1CCNC1=O)=O Cc1cc(=NC(=O)Cc2cccc(NC(=O)CCN3CCOCC3)c2)[nH][nH]1 N1(C(c2ccc(OC(F)F)nc2)=O)CC2CCCN(C(c3cnc(S)nc3)=O)C2C1 c1(OC)cc(N)c(C(=O)NC2C3N(C(=O)OC(C)(C)C)CC(CC3)C2)cc1F c1(C(=O)NC2(C)CN(C(C(C)Cc3ccncc3)=O)C2)cc2cc(Cl)ccn2n1 N1(C(c2cncc(C)c2)=O)CCC(NC(=O)CCOCC(F)F)CC(O)C1 C1(CC(c2nnnn2CC)Nc2scc(CC(=O)OCC)n2)CCC(C)(C)O1 c1(C(=O)O)ccccc1S(=O)(=O)CC(CN1C(=O)OC(CCCCS)C1=O)N(C)C c1(CNC(N2CC3C(Nc4cc(Sc5ccccc5)c[nH]4)C3C2)=O)ccccc1F C1(CC(=O)N(C2CCN(C(c3cc(-c4cccs4)[nH]n3)=O)C2)C)CCC(C)(C)C1 c1(C(N2CCC(O)(CCC)C2)=O)ccnc(C)c1O c1(C(N2CC3CC(NC(C4(O)COC4)=O)C2C3)=O)c(F)ccc(F)c1F Cc1cccc(CC(=O)N(CCC(C)NC(=O)C(F)n2cccn2)C)c1 c1(OC)cccc(C=CC(=O)NCC2CCCC(NC(c3n[nH]cc3C)=O)C2)c1 N1(CC(=O)N(C2C(C)CCNCC2)CCC2CC2)C(=O)c2ccccc2C1=O CN1N=CC(CS(=O)(=O)NCC(CC#N)NC(=O)OC(C)(C)C)C1=O n1(CC(C)C)[nH]c(CC(=O)NC2CCCCC2NC(c2cccnc2)=O)cc1=O c1(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)cc(C(N)=O)n(C)n1 c1(NC(C=CC(=O)NC(C(C)NC(=O)CC#N)C)=O)ccc(CN2CCCC2)o1 C(=O)(CC(C)(C)COC(C)=O)N1CCC(CNC(C#C)=O)C1c1ccccc1 C1(NC(C(C)NC(=O)OC(C)(C)C)=O)CCCN1C(C1CC1F)=O c1(C(=O)NCC2CCN(C(c3c(Cl)cc(C)s3)=O)C2)cc2cc(Cl)cnc2o1 N1(C(=O)OC)CC(C2CCN(C(=O)[O-])C2)C1 C1(O)(C(=O)NCC(C)CNC(=O)Cc2c[nH]nc2O)CCCC(C)(C)C1 c1(OC)ccc(CNC(=O)NC(CC2CC2)C(=O)O)cc1OC C1(CC(=O)N(CCN(C(C(C)NC(CC)=O)=O)C)C)COC(C)(C)CO1 c1(NC(N2CCC(NC(c3ccc(OC)o3)=O)C(C)C2)=O)c(C)cc(Cl)cc1Cl c1(CNC(CC2C(C)=NOC2=O)=O)c(C)nn2c1CN(C(=O)C=CC(C)C)CC2 C1(CNC(C2CCSCC2)=O)CCCCN1C(=O)CC12CCCC1C2 C1(C(N2CC3C(N(C(C4CC(OC)C4)=O)C)C3C2)=O)CCCCC1(F)F c1(C(N2C(CC)CN(Cc3ccc(Cl)nc3OC)CC2)=O)cc(C)c(O)c(C)c1 C12(CCNC(C3CC(=O)OC3)=O)CCC(CC1)N(C(=O)Cc1ccc(Cl)cc1)C2 C=C(C)C1OCCCC1C(=O)N(C)CCOCCNC(=O)C(C)(C)N(C)C N1(C(C2CCN(C(C)=O)C2)=O)CCCC2(CCN(C(c3cc(C)no3)=O)CC2)C1 C1(NC(C(C)CN(C)C)=O)CN(C(=O)CC(F)(F)Cl)CC12CCCC2 C(C)(C)(CC(=O)N1CCC(C(=O)Nc2cccc(Cl)c2)C1C)OC CCC(C)C(C)CNC(C1CCN(S(=O)(=O)Cc2ccccc2OC)CC1)=O CC1CN(C(=O)CCc2cscc2Br)CCC1NC(c1nccnc1N)=O c1(C(N2CC3C(NC(C(C=C)CC)=O)(C3)C2)=O)ncnc(C)c1C c1(SC)c(C(=O)NCC(O)CNC(C2(O)CCOC2)=O)nnn1-c1ccccc1 c1(C(=O)NC2C(NC(C(=O)Nc3ccc(OC)cc3)=O)C2)nccc(C)c1F C(=O)(CC(=O)NCCN(C)C(c1cc[nH]c1)=O)OCCC(C)C c1(NC(C2CC2CNC(C2CCO2)=O)=O)ccc(-c2cnccn2)cn1 C(C(C)(CC)C(=O)N1CC2(CC2)CC1C)NC(CNC(CCCCC)=O)=O C1(NC(C(N(OC)C)=O)=O)CN(C(C)=O)CC12COC2 Cc1cnc(NC(C2CN(C(c3ccc(CN=[N+]=[N-])o3)=O)C2)C)nc1 N1(C(=O)NCc2cccc(OCC)c2)CCC(F)(F)C(CNC)C1 c1(C(=O)NC2(c3nccs3)CN(C(COCCCC)=O)C2)cc(CC)nn1C CC(CC(=O)N1CC2CCCC1C2c1cn(-c2cc[nH]c(=N)c2)nn1)C(C)(C)C C1(C(=O)OC)COCC(C)(C)N1C(c1sncc1Br)=O c1(C(=O)NCCC(=O)NCC(C)(O)CNC(=O)C(F)F)ccccc1Cl Cc1ocnc1CNC(=O)CCC1(NC(=O)C=Cc2cocn2)CCCC1 c1(CC(=O)NCC(=C2CN(C(C(C)OC3CCCC3)=O)C2)F)ccccc1CO N1(C(C(c2cn(C)nc2)O)=O)CCOC(C)(CNC(C2(NC(N)=O)CC2)=O)C1 N1(C(C(N2CCSCC2)C)=O)CC2(CCC(C(=O)Nc3cc(CO)n(C)n3)O2)C1 C1(C(N(C2CCN(c3nccc(N4CCOCC4)n3)C2C)CC)=O)CCCC1(F)F CCC(C)CCC(=O)NC1CCN(C(C2CC2c2cncs2)=O)CC1 N1(C(C2C(C(F)(F)F)CC(=O)N2)=O)CC2CCCC1C2CNC(=O)CCC(F)F C1(C(C)CNC(=O)C(c2cccnc2)C)CCN(C(=O)C2=NOCC2)CC1 c1(CC)ncsc1C(=O)NC(c1ccccc1)C(C)NC(=O)Cc1n[nH]c(=N)s1 C1(NC(Cc2c(C)ccs2)=O)CCC(C)(C)CC1CNC(=O)C1=C(Cl)CCOC1 O=C(CCCC(F)F)NC1(CO)CN(C(=O)C2=NOCC2)C1 c1(CN2CC(F)(C(=O)NCC3CCN(CC)C3)C2)c[nH]c2cccnc12 CC(C)C(C(=O)NCCc1cccc(O)c1)NC(c1cnsc1)=O N1(C(CCCC#C)=O)CCC(C(=O)N(C2COCC2OC)C)CC1(C)C N1(C(c2c(C)cccc2)=O)CCC(NC(C2(c3ccno3)CC2)=O)C(O)C1 C12(NC(c3cccc(-n4cc(-c5cscn5)nn4)c3)=O)CCC(CC1)C2 N1(C(CCCCN(C(c2c(C)cc(N)cn2)=O)C)=O)CCOC2CCCCC12 C(=O)(C(C)CC(C)C)NCCCNC(c1c(CC)occ1)=O c1(C(N2C(C(=O)NCC3CCCC4CC34)CCC(C)C2)=O)ncc2ccccn12 O(NC(=O)C1=CC2(CN(C(=O)C(C)CC=C)C2)OC1)CCC#C c1(C(N(CCNC(CNC(=O)NC)=O)C)=O)cc2cc(Br)cn2c(O)n1 C(=O)(C#CC(C)(C)O)NC(CC1C(C(C)C)C1)=O.N12CCN(CC1)CC1CN2C1 n1(CC(=O)NCC23CCC2CCN3C(c2csc(CO)n2)=O)ccc(O)nc1=O c1(C(N2CCC(NC(c3[nH]cc(CC)c3)=O)(COC)C2)=O)cc(F)cc(N)c1F CCC(CC(=O)N1CCN(C(=O)Cc2sc(C)nc2C)CC(O)C1)C(C)C N1(C(C2C(CC)OCC2)=O)CC=C(CNC(c2csc(C)n2)=O)CC1 C=C(C)C1OCCC1C(=O)NC(C(=O)N1CCC(n2cncn2)C1)C(C)OC c1(C(N2CC(C)(NC(Cc3nc(C(C)C)sc3)=O)C2)=O)ccc([N+](=O)[O-])o1 CC1(CNC(=O)C(C)(C)CCF)CCN(C(c2cc(C(F)F)cc(F)c2)=O)CC1 CC(C)(CCCNC(=O)C(C)(C)C1CCOCC1)NC(C1CC2CC2C1)=O c1(CC)noc(CNC(=O)C(c2ccccn2)NC(=O)OC)n1 C1(CNC(CSC(C)C)=O)COCCN1C(=O)CNC(c1ccccn1)=O CC1CN(C(c2cnc(C3CC3)s2)=O)CC(C)C1NC(C12COCC(C1)C2)=O c1(C(=O)NCC(CN(C(c2c(CC)c(C)sc2)=O)C)O)c[nH]c2ccc(O)cc12 c1(CC)cc([N+](=O)[O-])ccc1C(N1CC(NC(=O)CNC(=O)C2CC2)C(C)C1)=O C#Cc1cc(C(N2CC(C)C(C)(CNC(=O)CC(=O)OC)C2)=O)ccc1C c1(C(c2n(CCOCC)nnn2)NCCc2c(Br)n[nH]c2Br)ccc(Cl)c(Cl)c1 c1(C(=O)NC(C(=O)NC(C#C)C2CC2)(C)C)ncc(C)cn1 C1(CC)COCC1NC(=O)C(CC1CCOCC1)NC(C1(c2ccno2)CC1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CCN(C(c2ccncc2C2CC2)=O)CC1)C Cc1nc(C(=O)NC(C(=O)NC2CC(O)C(O)C2)C2CC2)ccc1C#N C1(NC(C2CCCO2)=O)CCCC12CN(C(c1cc(-c3ccncc3)on1)=O)C2 Cc1cc(C)nc(CC(=O)NCC2CCN(C(=O)C(C)NC(N)=O)CC2O)n1 C(N=c1nc(N2CCC(C(O)C(N)=O)CC2)c2ncn(C)c2[nH]1)c1c(C)c[nH]n1 c1(NC(=O)Cc2ccc(F)cc2)ccc(-c2cccnc2)cc1 C1(NC(C2C(n3cc(CCN(CC)CC)nn3)CCC2)=O)CCCCCC1(C)C c1(CN2CCC(NC(C(C)c3ccco3)=O)CC2C)ccc(C#N)cc1F CCC(COC)C(=O)N1CCCCC1CCC(N1CC(F)(F)C1C1CC1)=O C1(CCC(=O)NC(C2N(C(c3ccc(C(C)=O)o3)=O)CCC2)C)CCC(O)CC1 C1(C(=O)NCCC2CCN(C(=O)CC3(CO)CC3)CC2)CCCCC1(F)F Cc1nc(NC(C)CCC(C)(C)C)cc(=NC(C)c2cc(N(C)C)n[nH]2)[nH]1 N(C1CCCn2nccc21)c1c(C(=O)NCCC2CCCO2)cccn1 c1(NC2CCC(CNC(c3cncs3)=O)CC2)nccc2occc12 C1(OC)CCCN(C(=O)C(F)CC(C)(C)NC(C2CC2C(N)=O)=O)C1C C(=O)(C(C)(C)Cn1ccc(SC2CC2)n1)NCC1C(NC(C=CCC)=O)C1 C1(NC(C(C)OCOC)=O)CC2(CCCCN2C(c2cnc3[nH]ccc3n2)=O)C1 N1(C(c2cc(NC(=O)C3CC3)c(Br)cc2)=O)CCC(O)CC1(C)C(N)=O.CCC N1(C(c2ccn(CCCC)n2)=O)CCC(NC(c2ccc(O)nc2Cl)=O)C1(C)C Cc1cc(C)c(NC(=O)C(c2ccc(Cl)cc2)N(C)Cc2csc(C)n2)c(C)c1 C1(C(=O)NCC)CCC(Cc2c(OC)cccn2)(NC(C23CCCC2C3)=O)CC1 Cc1ccc(C(N2CC3CC2C3NC(C2CCC(C)O2)=O)=O)c(C(C)C)n1 C1(CC(=O)NC)CN(C(=O)C(C)NC(C2CCCCCC2)=O)CCN1C(=O)CO S(=O)(=O)(c1ccc(C(N2CCCC(n3cncn3)C2)=O)cc1)NC(C)(C)C Cn1cc(CCNC(c2sccc2NCc2cncs2)=O)c2ccccc12 C(N=c1nc2c(cnn2C)c(NC2CC23CCC(O)CC3)[nH]1)C1CC(=C)C1 CC(CC(=O)N1CC2(CC(C(=O)NC(CO)C3(O)CC3)C2)C1)C(F)F c1(C(=O)NC(c2cccnc2)C(=O)NC(c2cscn2)C)cccc(F)n1 C(=O)(CCS(C)=O)NCCN1CCC(NC(c2ccc(CCC)s2)=O)C1 n1(CCCNC(C2CCN(S(=O)(=O)C3CC3)C2)=O)cc(CO)nn1 c1(C(=O)NCCCOCCCNC(c2ccn(CC)n2)=O)cccc(=O)n1C C(=O)(C1=COCCO1)NC(C1CCCCC1)CNC(c1ccc(OC)s1)=O C1(NC(c2ccc(CC)nc2)=O)CN(C(C2CSCN2CC)=O)C2CCCCC12 O=C1CCC(CCC(N2CC3C(NC(C4(C5CCC5)CC4)=O)C3C2)=O)CN1 c1(NC2(CCOC)CCC2)ncnc(NC(C2CCOC2)COC)c1C c1(N(CCNC(=O)CCC2CCCC(=O)N2)CC)ncc(C#N)cc1Cl C1(C(N(CCN(C(C)C)C(c2cnc(S)nc2)=O)C)=O)CCCC(=O)CC1 S(=O)(=O)(c1cccnc1NCc1ncsc1C)NC(c1ccccc1Cl)CC Cc1nc(C)c(C(=O)NC23CC(NC(C4CCN(C(=O)C5CC5)C4)=O)(C2)C3)s1.OC C1(C)(C(=O)NCC(CN(C(C)C(=O)NC2CCCCC2)C)CO)CC2(CC2)C1 Cn1c(C(N2CCCC(CNC(C3Cc4nnsc4S3)=O)C2)=O)cccc1=O N1(C(C(c2cc(F)cc(F)c2)=O)=O)CCCC2(CCN(C(C3(O)CC3)=O)C2)C1 CN1CCOCC1CC(=O)N(C1CCN(C(=O)C=C(Cl)Cl)C1)CCO C(C)(CCC(=O)NCC1CC(NC(C2(F)CCCC2)=O)C1)OCC c1(C(=O)NCC2C3CN(C(C(CC)=CCCC)=O)CC32)cc2sc(C)nc2[nH]1 c1(CC(=O)NC(C)(CNC(C2OCC2(C)C)=O)C2CCC2)ccc(F)c(Cl)c1F c1(C(=O)NC(CN(C(=O)C(C)C(C)(C)C)CC)C)ccc(Cl)c(F)c1N N1(C(C(C)CO)=O)CC(NC(c2ccc(P(C)(C)=O)cc2)=O)Cc2ccccc21 c1(N2CC(C(N(C3CCNC3)C)=O)CC(F)(F)C2)ncnc2ccc(I)cc12 Cc1cc2cc(C(=O)NC3CCCC3NC(c3cn(C)[nH]c3=N)=O)c(Cl)cc2[nH]1 N1(C(C2C(C(=O)OC(C)(C)C)C2)=O)CC2CC3CC2C1C3NC(=O)C1=CCC1 CC1C(NC(C2CC23CCC3)=O)C(C)CCN1C(=O)Cn1cc(C2CC2)nn1 C1(NC(c2ccc(F)c(O)c2)=O)CCC(O)CN(C(=O)C(F)C2CCC2)C1 n1(CC)cc(CC(N2CC(N(C(=O)CNc3ccccn3)C)C2)=O)cn1 N1(C(c2ccc(CC)cc2)=O)CCCC2(CCN(C(=O)CCC(C)OC)C2)C1 c1(C(=O)NCCC2OCCN(C(C(C)CF)=O)C2)cc(Cl)cc2ccncc12 N1(C(c2c(OC)cc(C)s2)=O)CC(NC(=O)CSc2ccccc2)CC12CCC2 C1(NC(CNC(=O)NC)=O)CCCCCC1C(N1CC(O)C(O)C1CO)=O O=C1CC2CCCC2(C(N2CCOC(CNC(c3cc(C(F)F)[nH]n3)=O)C2)=O)C1 c1(C(N2CC3C(C(=O)Nc4cccc(C(C)C)c4)(C3)C2)=O)c(Cl)cc(Br)cc1Cl C1(NC(c2cc(C)oc2)=O)COC2(C1)CN(C(=O)C(O)CC1CC1)C2 C(=O)(C(O)CNC(=O)C=CC(C)NC(c1cc(C(C)C)[nH]n1)=O)NC n1(COCC)nnc(C(=O)NCCCNC(=O)CCCc2cccc(Cl)c2)c1N c1(C(N2CCC(C)(NC(C3(OCC)CCCC3)=O)C2)=O)ccnc(F)c1N N1(C(=O)Cc2cc[nH]c2)CCC2C(CCCN2C(C2CS(=O)(=O)C2)=O)C1 C(C(CC1CC1)C(=O)N1CCOC(C(N)=O)C1)NC(C1(COCC)CC(=C)C1)=O N1(C(c2nccs2)C)CCN(c2ccc(CN)cn2)CC1 CN1CCCC(N(C=Cc2cncn2C)CCCO)C1=O c1(C(=O)NC2C=CC(NC(c3ccc(CCC)cc3)=O)C2)cccc(Br)c1O C1(Nc2cc(N3CCC(CC)OCC3)nc(C)n2)CCCC(C2CC2)C1 C(=O)(CCC(=O)NN(C)C)N1C(C(N(CCO)CC)=O)C(C)C1 C(=O)(CCC(C)(F)F)N(CCC(=O)NCCC(=O)OCC)CCO CC(C)CS(=O)(=O)CC(=O)NCC1(F)COCCN(C(=O)C(=O)NCC2CC2)C1 c1(C(N(C)CC2N(C(Cc3cc(C)ns3)=O)CCOC2)=O)cnn2ccccc12 C(CCCCC(=O)NC1CC1CNC(c1ccc(F)c(Cl)c1)=O)NC(N)=O CC1(C)CN(C(=O)CCP(C)(C)=O)CC1CC(=O)NCCC1CCCC1 C1(C#CC(=O)N(C)CCNC(c2cc(N)c(O)c(F)c2)=O)(CC)COC1 c1(-n2c(NC(=O)NC3CCCC3N3CCOCC3)ncn2)cccc(F)c1 C1(CCCC(=O)N(C2CCN(C(=O)CC(C)(C)C)C2)C)CCCC(=O)N1 C1(C(=O)NCC(C(C)C)(C)O)CC(F)(F)CN1C(c1cc(O)cc(F)c1)=O C1(NC(c2cncc(COC)c2)=O)COCCN(C(C2(O)CCC2)=O)C1 C1(C(N2CC(OC(=N)O)C2)=O)CCCCN1C(c1c(C)cco1)=O C1(C(=O)NCc2ccc(CCNC(CCCC=C)=O)cc2)CCCCC1N=[N+]=[N-] C1(CC=C)(NC(C2CC(=O)N(C)C2)=O)CCCN(C(c2ccnnc2O)=O)C1 C(C(C)(C)CNC(C1CCOC1CC)=O)N(C(C1(CC=C)CC1)=O)C c1(C(=O)NCC2CC(CNC(COCCC)=O)OC2)ccc(C2CC2)cc1F C1(C(N(C)CC2CCN(C(=O)C=CC3CCCO3)C2)=O)C2CC3C(C2=O)C13 C(C(COC)C(=O)NC(C1CC(NC(=O)CCc2cccn2C)C1)C)OC C1(NC(C2N(C(C(C)=C3CC3)=O)C3(CC2)CC3)=O)CCN(C)CC1C#N C1(C(=O)NCCCCNC(CCc2c(C(=O)OC)nco2)=O)CCCCC1C CN1CCN(C(C2C3CCC(C3)C2C(F)(F)F)=O)C(=O)C1 C1(NC(c2cc(Cl)cc(Cl)n2)=O)CCCN(C(=O)COC2CCCC2)CC1 N1(C(C2C(C)(C)CC(=O)N2)=O)CCCC(C2(NC(C3CSCCS3)=O)CC2)C1 C#Cc1ccc(Cl)c(C(=O)NCCOC2CN(C(C3(O)CCSCC3)=O)C2)c1 c1(C(N(C2CCN(C(=O)CC3(O)CCCOC3)CC2)CCC)=O)nc(C)c(C)o1 CC(C)CC(CNC(C1CC(=O)N(C)C1)=O)NC(C1CC=CC1)=O C12(C(N3CC(NC(C(CC)Br)=O)(CO)C3)=O)CCCCC(=O)N1CCC2 N1(C(C2(CC)CC2)=O)CCC2(CC1)CC2CNC(=O)CC1CNC(=O)C1 C1(C(N2CCCC(CC)(CO)C2)=O)N(C(=O)C(C)N=[N+]=[N-])CC12CCCC2 c1(CC)cc(F)c(C(=O)NC(C)C(C)NC(c2n[nH]c3c2COCC3)=O)cc1F N1(C(C(C)C2CCOC2)=O)C(C(=O)N(C)Cc2cc[nH]n2)CCC12CC2 C1(CC)CN(C(=O)C(=O)NC2(c3cccc(C)c3)CC2)CCN1C(C)C C12(CNC(Cc3c(C)nsc3)=O)CCC(CC1n1cc(C(C)(C)O)nn1)C2 c1(OC)cc(OC)c(C(=O)NC2CCCC2NC(=O)CCCCC2CC2)cc1N CC1CCN(C(=O)CCCn2ccnc2)CC1NC(=O)C(c1cnn(C)c1)=O C#CCCC(=O)NNc1cccc(Cl)c1-c1ccc(OC)cc1 c1(CC(=O)NCC2C(CNC(C3(C)CC(F)C3)=O)C2)ccc2occc2c1 C1(CC(=O)NC2CCCCN(C(=O)C=Cc3cncs3)C2)CCC2(CC1)CC2 N1(C(C2CC(=O)NCC2)=O)CC2CCN(C(c3ncc(Br)cn3)=O)C2C1 c1(-c2cc(N(C(=O)C=CC(F)F)C)[nH]n2)cccc(Cl)c1 N1(C(C2(CC#C)CCCOC2)=O)CCCC(O)(CN(C(=O)CCP(C)(C)=O)C)C1 CON(CC1CCCC(C)C1)C(=O)NC1(c2ccoc2)CC1 c1(CC(=O)NCC2CCN(C(c3cnc(OC)s3)=O)C2)cc(O)nc(O)n1 c1(C(=O)NCC2C(NC(Cc3c(OC)ccc(F)c3)=O)C2)cccc2[nH]ncc12 Cc1cncc(CCNC(=O)C(C)CC2CCCO2)c1 C1(NC(CN(c2ncccn2)C)=O)CCN(C(c2cccc(Br)c2)=O)C1(C)C Cn1nc(C(=O)NCC2(F)CCN(C(C3(C)COCCO3)=O)C2)cc1C(C)(C)C N1(C(c2cc(COC)no2)C(=O)NCCCOC)CCN(C)C(C)C1 Cc1ccc(O)c(NC(=O)CC2CN(C(=O)CCc3cnoc3)CC2C)c1 S(=O)(=O)(c1ccc(NCC2CCN(C(c3cc(C#N)ccc3C)=O)C2)cc1)NC N1(C(CSCC(C)C)=O)CCC2(CC1)CN(C(=O)C(F)(F)CC1CC1)C2 CC1CN(C(=O)CCCc2ccsc2)CCCN1C(=O)COC1CCCC1 Cc1cc(C)n(CCCC(=O)NNC(=O)c2cccc(N)n2)n1 N12CCN(CC1)C(=O)C2.c1(NC(C)=O)ccc(C(=O)N(C)CCOC(F)F)o1 c1(C(=O)NCCN(CCC)C(c2ccc(C3CC3C)o2)=O)ccc2nsnc2c1 N1(C(C(CC)OC)=O)CCC2(CCCC2NC(c2cc3c(ccn3C)s2)=O)CC1 c1(CNC(CCCN(C(=O)CCC(C)N(C)C)C)=O)ccc(F)c(F)c1 CCC(C)CC(=O)C(=O)NC(C1CN(C(=O)CCn2cc(C)cn2)C1)C S(=O)(=O)(CC(=O)NC1(C(=O)NCCCN2CC=CC2)CC1(C)C)NC O=C(C1=CCC2(COC2)OC1)NCC=CCNC(c1nccc2occc12)=O C(=O)(CC(C(C)OC)NC(c1ccc(C(C)=O)o1)=O)NCCC(CC)(C)C N1(C(C(C)C2CCOC2)=O)CCC2(CCCN2C(=O)Cc2csnn2)C1 c1(C(=O)NCCC2(O)CN(C(c3cc(CCC)on3)=O)C2)cnn(C)c1CC CCCC(CCC)C(=O)N1CCC(CCC(N2CCC(O)C(CC)C2)=O)C1 CC1CSCCN1C(C1CCCC(NC(=O)C(=O)NCC(F)F)C1)=O c1(CC(=O)NCCN(C(=O)COc2cn[nH]c2)CCOC)ccccc1C1CC1 c1(C(N2CC3C(CNC(COC)=O)(C3)C2)=O)cccc(C)c1N c1(CCNC(=O)NCCC=CCCC)csc(-c2ccccc2)n1 c1(CC(=O)NCCC(O)CNC(=O)C=CC2CCOC2)ccccc1Br C(=O)(CS(C)(=O)=O)NCC1N(C(C(N2CCOCC2)C)=O)CC1 C1(NC(C2(CF)CCN(C(c3nn(C)c(CO)c3)=O)C2)=O)CC(O)CC(C)(C)C1 c1(CC)ccc(F)cc1NC(C1(CNCc2cc(O)cc(Br)c2)CC1)=O C1(CC(=O)NCCC2(NC(=O)C(O)CC3CCOCC3)CC2)(COC)CCCC1 C1(CNC(c2ccc(C(F)F)s2)=O)C2CN(C(C3CCN3C3CCCC3)=O)CC12 C(CCCCC(=O)N(CCC1CN(C(c2c(C)nsc2N)=O)C1)C1CCC1)NC(=O)OC c1(C(=O)NC2CCC(CCNC(CCCSC)=O)C2)cnc2ccnn2c1N c1(SCC)ccc(OC)cc1C1N2CC(C(SC)C2)N(CC)CCNC1=O.S(C)CO C1(NC(c2c(Cl)ccc(C)c2)=O)CC2CCC1CN2C(C1(CC2CC2)CC1)=O CCC(O)C(C)(C)C(=O)N1CCCCC(N(C)C(c2ccnc(C)c2C)=O)C1 N1(C(c2ccncn2)=O)CCC2CCCC(C1)N2C(c1cnc(Cl)s1)=O c1(OC)ccccc1CNC(=O)COC1CCN(C(c2c(OC)noc2C)=O)C1 Nc1cc(C(N2CCN(C(=O)CSCC(F)F)CC2CO)=O)nc2ccccc12 C1(CNC(=O)NC(c2cn(CCCF)nn2)C)CCCCC1(C)C N1(C(C(C)c2ccco2)=O)CC(NC(=O)Cc2csc(Br)n2)CC2(CC2)C1 Cc1nc2cccc(C(N3CC(CNC(c4cc5nc(C)sc5[nH]4)=O)C3)=O)c2[nH]1 C1(CN(C)C(c2cnc(Cl)s2)=O)CN(C(C2COC(=O)O2)=O)CCO1 N1(CC)CCN(C(=O)NC(c2nc(C)no2)C)C(C)C1 c1(C(=O)NC(CC)C(=O)NC(C2CCC2)C)cc(O)cc(F)c1 c1(CN(C(=O)CCN(C(C2CC=CCO2)=O)C2CC2)C)cccnc1O N1(C(C(C)OCCC=C)=O)C(CNC(c2ccn(C)c(=O)c2)=O)CC2CCCC12 c1(C(=O)NC2(CC=C)CCN(C(c3cc(C)on3)=O)CC2)nc(O)nc(O)c1N C12(CC(c3ccc(Cl)o3)=O)CC(C1)C(NC(c1nccc(C(=O)OC)c1)=O)CO2 c1(C(=O)NC2C(NC(c3ccc(C#N)cc3)=O)CCCC2)ccc2n[nH]cc2c1 N1(C(C23N(C(COCCCCCC)=O)CC(C2)C3)=O)CCc2c[nH]nc2C1 c1(N(C(=O)OC(C)(C)C)C(N)=O)ccc(F)cc1O.Cn1c2cnc1SC2 C=C1CCC(C(=O)NC2CN(C(=O)C=CCF)CC2C(F)(F)F)CC1 C(=O)(CC(COC)CNC(=O)CCc1ccc(C)cc1C)NC C(=O)(N=c1cnn(C)[nH]1)C1CCC(NS(CC=C)(=O)=O)CC1 c1(C(=O)NCC2C(CNC(CCOC(C)C)=O)C2)cccc2cncn12 C1(C(NOCCCC#C)=O)CC(C)CN(C(=O)C=Cc2ccnn2C)C1 CCC(CSC)N=c1ccnc(N2CCC(c3c[nH]c(=N)[nH]3)CC2)[nH]1 C1(C)(CNC(c2nc(C)sc2C)=O)CN(C(=O)CC2(N3CCCC3)CC2)CCO1 C1(C(=O)NC(C=C)C2CC2)CC2C=CC1C21CC1 c1(SC(C)C(=O)N2CC(N(C(=O)C(O)c3ccco3)C)C2)ccc(F)cc1 C#Cc1ccc(C(N2CC(CNC(=O)CCCc3nc(C)cs3)CC2C)=O)cc1 C1(NC(c2cccc(OCC)c2)=O)C2CC1CN(C(C1CC13CCCOC3)=O)C2 c1(N2C(C)CC(NC(c3c(CCC)nco3)=O)C2)cc(C)c([N+](=O)[O-])cc1F C1(NC(C2CNC(=O)N2)=O)CCCCC1CNC(c1ccsc1)=O CC1CN(C(=O)Nc2nn[nH]c2C(F)(F)F)CC1CCSc1ccccc1 c1(CN(C(CC=CC=C)=O)C)cccc(CNC(C2COC(=O)N2C)=O)c1 C1(OCC)CCN(C(=O)C=CCN(C)C(C2CCN(OC)CC2)=O)CC1C c1(OC)nc(C)ncc1C(=O)N(CCNC(C1CN(C)C(=O)N1)=O)C1CC1 C1(N(C(CC2ON=C(C)C2)=O)C)CC2CC1N(C(c1nc(O)c(C)s1)=O)C2 C(C(C)C(C)C(=O)NCc1cc(C(=O)Nc2c(CO)cccc2F)co1)OC c1(NCc2n(CCC)ncn2)ccc(N(C)C)cc1 c1(SCC2CC2)cnc2c(c1)COC2.c1(OC)ccc(C(=O)C(=O)N)cc1.O CC(CN(C)C(c1cc(CNC(=O)C(C2CC2)C2CC2)no1)=O)C(C)(C)C c1(C(=O)NCC=CCNC(=O)CC2CC2(Cl)Cl)cccc(OC(F)(F)F)c1 N1(C(C2CCN(C(=O)OC)CC2)=O)C2CCC1C(C)C(NC(C1CC1C)=O)C2 CN1N=C(C(=O)NCC2C=CCN2C(c2cc3c(O)cccc3[nH]2)=O)CCC1=O c1(C(N2CCC(C)(NC(C(F)=C(C)C)=O)C2)=O)ccc([N+](=O)[O-])cc1Br c1(-c2ccc(CC(CC)C(=O)NS(C)(=O)=O)cc2)ccc2c(c1)C(C)C(C)O2 CC1=C(C(=O)NC(CCN(C)C)C(=O)NC2CCCN(O)C2=O)COCC1 Cn1cc(C(N2CCN(C(=O)C(F)C3CCC3)CC2CO)=O)c2ccccc12 N1(C(c2cnc(SC)s2)=O)CC2(C1)CN(C(=O)CCN1CCCC1=O)CC2CO CCS(=O)CC(=O)N1CC=CC1(C(=O)NCCc1nc[nH]n1)COC C1(C(=O)NC2(CC=C)CN(C(c3[nH]nnc3C)=O)C2)C(Cl)(Cl)C12CC2 Cc1cccc2c1OC(C(=O)NCC1CN(C(=O)C=CC3CCCC3)CC1C)C2 CC(Cc1ccco1)C(=O)NCC(=C1CN(C(c2ccsc2)=O)C1)F N1(C(Cc2c(CC)con2)=O)CC2(COC(CNC(=O)CNC(N)=O)C2)C1 N1(C(CCN(C(COCCCCC)=O)CCCO)=O)CCC(C)(C)CC1 C1(NC(CSCC#C)=O)CCC(NC(C2CCN(S(C)(=O)=O)C2)=O)C1 C(=O)(CC(C)C(=O)NCC(c1ccco1)NC(C1(CCF)CC1)=O)OC N1(C(c2c(NC)cncc2)=O)CCCC12CCN(C(=O)CN=[N+]=[N-])C2 N1(C(C(CCC)OCC)=O)CC2CC(C)N(C(c3cn(C(C)C)cn3)=O)C2C1 c1(C(N2CCC(CC=C)(NC(C3COCCN3C)=O)C2)=O)nc(C)ccc1F C(C(C)S(=O)(=O)c1ccccc1)NC1COc2c(C)cccc2C1 O(N1CCC(CC(=O)NCC(CNC(=O)C(O)CCSC)CO)CC1)CC C1(C(C)C)(CO)CCN(C(C2CCN(C(c3cc(Cl)n[nH]3)=O)C2)=O)C1 C=CCCCCC(=O)N(C(CNC(c1cnn(CCO)c1C)=O)CC)C c1(C(=O)NC(C2CC(NC(c3cc(OC)n(C)n3)=O)C2)C)cccc2oncc12 c1(C(=O)NCC(C2CC2)NC(C2(CC=C)CC=CC2)=O)ccc2c(c1)ncn2C c1(SC)ccc(C(N2CC3CN(Cc4c(CC)cccc4)C3C2)=O)cc1Br c1(CNC(CCC=C)=O)cccc2c1CCN(C(=O)C(C)(C)c1nccs1)C2 N1(C(C(C(C)NC(CCOC)=O)(C)C)=O)CC2(C1)OC(=O)NC2C c1(CCC)nc(C)c(C(=O)NC2CCN(C(C3CCCN(CC)C3)=O)C2C)o1 N1(C(C(c2n(C)cnc2)O)=O)CCC(C)(NC(=O)CCC2CC(F)(F)C2)CC1 c1(N2C(NC(C(C=CCCC)O)=O)C(C)CC2)cc2nncn2cn1 CC1(C)CN(C(c2ccc3c(c2)OCC3)=O)CCC1NC(=O)CCSCC(N)=O c1(C(=O)NCC(CNC(=O)CCc2ncccn2)OC)ccc(Cl)nc1 C1(CC)C(NC(c2csc(Cl)c2)=O)CCN1C(c1cc(Cl)cn1C)=O Cc1ncc(Br)c(C(N2CCOCC2CNC(C2(CO)CC2(F)F)=O)=O)n1 C1(C(=O)O)(COC)CC(=O)C1.c1(C(CN(C(=O)C(CO)N(C)C)CC)O)ccccc1 C(=O)(C1=C(C)CCOC1)NC(C)(C(OC)OC)CC.C=C1CC2(C1)C(=O)NC2 CCCC(C(=O)N1CCCC(CF)C1)NC(c1cnc(OC)nc1)=O O=C(CC(C(F)(F)F)N1CCOCC1)N1CCC(C(=O)Nc2cncc(F)c2)C1 C12(NC(c3cc(COC)c(C)s3)=O)CCCC1N(C(=O)CNC(=O)C1CC1)CC2 C(=O)(C#CC(C)(C)C)NCC(CC)NC(=O)CCCn1ccccc1=O CC1CN(C(c2cc(N)cnc2Br)=O)CCC1NC(=O)CC(F)(F)F C1(CNC(c2cc(C)c(C)s2)=O)CCC2(CO1)CC(NC(C1CCCS1)=O)C2 C1(CNC(CNC(CNC(CN(C)C2CC2)=O)=O)=O)CCC1(C)C c1(C(N(C)CC2CCN(C(C3C(C)C3)=O)C2)=O)cccc2c1OC(F)(F)O2 C1(CN(C(C(n2c(C)ncc2)C)=O)C)CCCN(C(=O)CCc2ccco2)C1 N1(C(c2c(C)ocn2)=O)CC2CC(NC(=O)C(C(C)C)n3cnnc3)CC2C1 c1(C(C(=O)NC(CNC(C2C(C(=O)OC)C=C2)=O)C)(F)F)ccc(C#C)cc1 C1(C(N2CCC(OCCNC(CCNC(C)=O)=O)CC2)=O)CCCC(C)(C)CC1 Cc1noc(C)c1CC(N1CC(NC(c2ccnc(OC(C)C)c2)=O)C(C)C1)=O CC12COC(C(=O)NC3CCN(C(c4cccn4C4CC4)=O)C3C3CC3)(C1)C2 C(=O)(C(C)C(F)(F)C(F)F)N1CCC(C)(NC(C2(CC=C)CCOCC2)=O)C1 N1(C(c2cncc(N)c2)=O)CCOC2(CCCN(C(=O)C(O)CC(F)(F)F)C2)C1 C1(C(=O)NCC(=C2CCCN2C(c2ccc(C)c(O)n2)=O)C)CCOC(=O)CC1 c1(C(N2CCC3(NC(CC4(C)CC4)=O)C(C2)C3)=O)ccc(S(N)(=O)=O)c(F)c1 C1N=C(NCC)Nn2cc1cn2.C1(CO)CC2C=CC1O2.C(=O)(C)NC1CC1 c1(CC(C)NC(C2C(C(=O)OCC)C2)=O)ccccc1CC C1(NC(C2CCC(F)C2)=O)CC2CCC1CN(C(c1csc(=NC3CC3)[nH]1)=O)C2 c1(C(=O)NCC2N(C(C(C=C)O)=O)CC2)ncnc(C)c1C N1(c2cccc(C)c2)CCN(c2ccc(C#N)cn2)C(CCC2CC2)C1 C(=O)(CCCC(=O)NCC(C)CC(=O)NC1CNC(=O)C1(C)C)OC Cn1cc(C(N2CC(NC(c3cc[n+]([O-])cc3)=O)C(F)C2)=O)nc1O C1(NC(CCCOC)=O)CCCC(N(C)C(c2nc(Cl)cs2)=O)C1 c1(OCC=C)ccccc1C(=O)NC1CC(CCO)C1.C12CCN(C1)C(=O)CO2 C(CC(C(=O)Nc1nc(CC2CC2)no1)N1CCOCC1)NC(=O)OC(C)(C)C N1(C(C(CC(C)C)O)=O)CCC(CCNC(=O)C(=O)NCC(F)F)C(F)(F)C1 C1(C(C(=O)NC2CC(NC(CCC3CC(OC)C3)=O)C2)C)CCC(C)(C)CC1 N1(C(C(C(C)(C)O)NC(C2CC(=C3CCC3)C2)=O)=O)CCN2CCCCC1C2 C1(CNC(C2C(c3c(C)c[nH]n3)C2)=O)CC2(CO1)CN(C(c1cc(C#N)on1)=O)C2 C(=O)(C(C)CNC(C1(CC)COC1)=O)NC(C#C)CC N1(C(C2(c3cccc(C(=O)O)c3)CC2)=O)CCC(NC(C2(O)CC2)=O)CC1.CCO N1(C(c2ccc(OC)s2)=O)CC(NC(c2[nH]c(C)nc2C)=O)CC12CCCC2 n1(CC(=O)NC2CN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)ncccc1=O C1(C(N2CC(NC(CC(C(C)C)(F)F)=O)C2)=O)CC2CS(=O)(=O)CC(C1)C2(F)F c1(CC(N2CC(COC)(NC(=O)CCC3CC3(Cl)Cl)C2)=O)cc(C2CC2)nn1C c1(COC(=O)NCCn2cc(CCC(C)O)nn2)c(C(F)(F)F)noc1C N1(C(c2cnn(C)n2)=O)CCCCCC1C(=O)Nc1cncc(Cl)c1 c1(C(=O)NC(C)CNC(=O)COCC(F)F)ccccc1OC(F)F.S(=O)(=O)(C1CC1)N C1(COC)(CNC(c2cnc(O)s2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1 c1(SC)cc(N2CCN(CC(C(CSCc3ccccc3Cl)=O)=O)CC2)ncn1 C12(CNC(C3(C)CC(F)(F)C3)=O)CC(CO1)N(C(c1cc(C(F)F)[nH]n1)=O)C2 C(=O)(C1=NN(C2CC2)C(=O)CC1)NCC1CC(NC(C(c2cccc(C)c2)O)=O)C1 CC(C)CC(O)C(=O)N1CCCC(CNC(=O)CCc2nc(O)n[nH]2)CC1 N1(C(C2CCC(CC(C)C)CC2)=O)CCN(C(=O)C(O)C2CCC2)C(CCO)C1 c1(CC)cc(C(=O)NCCCOCCN(C(=O)CCCNC(=O)OC)C)on1 N1(C(CN(C2CCC2)C(C)C)=O)CCC2CC2(C(=O)O)CC1.C1(N)CCCCC1C C1(CNC(C(CC)COC)=O)CCN(C(=O)CCc2cnoc2)CC1CC CC(C)(C#N)CCC(=O)NCCNC(c1ccc(C(F)(F)F)cc1)=O Cc1ccncc1CC(=O)NC1CCC1CNC(C1C2CCCC12)=O Cc1cc(C(=O)NC(C2CN(C(C3CCC(=O)C3)=O)C2)C)n(C2CC2)n1 CC(CCC(C)(C)C)C(=O)N1CC(C2CC2)(C(N2CC(C)CC(C)(C)C2)=O)C1 C1(NC(C=CC(CC)=CC)=O)CC2CCC1N2C(=O)Cc1cnc(C)o1 C(=O)(C1=C(c2ccccc2)SCCO1)N1CC(C)(CNC(C2CC(OC)C2)=O)C1 c1(C(C(=O)NC(C)C)N(C)CCOC(=O)C2CC2)cc(Br)sc1Br c1(N(C)CC2(OC)CCCOC2)ncc(I)c(C)n1 C(=O)(C1CCCc2sccc21)NC1C(NC(c2c(SC)cc(F)cc2)=O)COC1 c1(Cc2cnc(C(=O)OCc3nnc(CC)o3)s2)c(F)cccc1F c1(CN(C(CC)=O)C)nnc2n1CCN(C(C1C3C4CCC(C4)C13)=O)C2 N1(C(C2CCC(CC)O2)=O)CCC2(CCC2)C(CNC(C2(O)CC(C)(C)C2)=O)C1 N1(C(=O)NC(CC=C)Cc2ccccc2)CCc2c(C#N)cccc2C1 c1(CC(=O)NC(CN(C(c2c(OC)n[nH]c2)=O)C)C)ccc(F)c(Br)c1 C(CC(O)CC(=O)NCC#CCNC(C1CCC(=O)NC1)=O)SC C1(C(C)C(=O)NCCCn2ccnc2)CCN(C(C2CS(=O)C2)=O)C1 C1(CF)(N)CCN(C(c2snnc2C2CC2)=O)C1.CCCCCCNC(=O)CNC=O C(=O)(C(C(C)C1CC1)N(CCCc1ccco1)C)NCCOC c1(C(=O)NCC(CC)NC(c2cncc(N(C)C)c2)=O)cnc(O)c2ccsc12 c1(CC)cc(C(=O)NCC2(CNC(C3CCC(C)S3)=O)CC2)no1 c1(C(N2CC=CC(NC(C(C)OCCOC)=O)C2)=O)ccc2nc[nH]c2n1 C1(C2CC2)(C(=O)NC2CCC(CCNC(C3(C)CCC3)=O)C2)CCC1 C1(NC(CCOCCCOC)=O)CN(C(c2ccoc2)=O)C2(CCCOC2)C1 N1(C(C)=O)CCCN(C(C2CN(C(C3CCC3C(C)(C)C)=O)CC(C)O2)=O)CC1 C1(C(C)C)N(C(=O)Cn2ncnn2)CC12CCN(C(C1(C)CC3CC3C1)=O)CC2 C1(CCNC(C2(n3cccn3)CCCC2)=O)CCCN1C(=O)CC1CCCCC1 c1(C(N2CC(OC)(CNC(C3(C)C=CCC3)=O)C2)=O)cc(O)c2ccsc2c1 C1(CNC(CC(CN(C)C)(C)C)=O)CCC(C)(C)CN1C(=O)CC12CCCC1C2 Cc1nc2cc(Cl)ccc2n1CC(N1CCCC(NC(C2CCOCC2)=O)C1)=O C1(C(=O)NCC(C)(C)OCCNC(=O)C(F)F)CCN(c2ccc(Cl)cc2)C1=O N1(C(C2(OC)CCSC2)=O)CC2CC2(NC(=O)Cc2csc(C(F)(F)F)n2)C1 C(=O)(C1=CCC(F)(F)CC1)N1CC(C)C(CNC(c2ccc(=O)n(C)c2)=O)CC1 C#CCC(CC(=O)N(CCCCO)C)NC(=O)C(C)Cn1ccnc1 c1(C(=O)NC(c2ccc(OC(F)(F)F)cc2)C(=O)OC)c(I)ncn1C C1(F)(CNC(CCC(=O)N(C(C)C)C)=O)CCCN(C(C2COCC2(C)C)=O)C1 C1(CC(=O)N(C2CC=CC2)CC)C(NC(=O)Cc2cccs2)CC1O N1(C(CN(CCC)C)=O)CCC2(CC1)CC(NC(=O)C1=C(Cl)CCC1)CO2 C12(CNC(CCCC(=O)NC(C)C)=O)CN(C(=O)CC3=CCCC3)CC(F)(C1)C2 C1(C(=O)NCC2CC23CC3)(CC)CCCN1C(=O)CCCNC(C)=O n1(CC)ncc2cc(C(=O)NCCNC(=O)C(F)C3CCOC3)c(C)nc12 N1(C(c2c(C)cc(OC)nc2)=O)CC2=C(C1)CN(C(=O)Cc1cccc(Cl)c1)C2 Cc1cc(CNC(C2CCCN2c2nnn(C)n2)=O)on1 c1(C(N2C(c3cn(CCOCC)nn3)CCC2)=O)coc2c1CSC2 N1(C(=O)OC(C)(C)C)CCC(CCN2CCN(Cc3ccc(Cl)cc3)CC2)CC1 C1(CC)CCCC1(C)C(=O)NCC(C(C)C)NC(C1CCCN1C(C)(C)CC)=O CCCC(F)C(=O)NC1CC12CC(C(N1CC(c3nc(C)no3)C1)=O)C2 C1(O)(C(C)NC(c2cc(-c3ccsc3)[nH]n2)=O)CCN(C(=O)CNC(N)=O)CC1 c1(CN2CC3(CC(NS(=O)(=O)C(F)(F)F)C3)C2)cccc2c1OCO2 C1(C(=O)NC2C(C)(O)CCC2)CC2C=CC1N(C(C13CCC(CC1)C3)=O)C2 c1(C(=O)NC(CC(=O)NCC(C)(C)N(C)C)C(F)F)c[nH]c2ccccc12 C1(C(N(C)Cc2c(C)nn(C)c2)=O)CC(C)(C)CN1C(C1CC(=O)NC(=O)C1)=O c1(-c2cn(CCN(C(=O)C(C)(C)N3CCCC3)C)nn2)c(F)cc(F)c(F)c1F c1(C(=O)NCC2CC(C(=O)NC3CN(C)C3)C2)c(O)cccc1F C1(O)(CN(C)C(C2CCCS2)=O)CCCN(C(=O)CCn2cnc(=N)[nH]2)C1 C1(C(C)C)C(C(=O)NC2CC(O)C2O)CCN1C(c1c[nH]nc1Cl)=O N1(C(c2c(C(C)C)ncnc2)=O)CCN(C(=O)C(c2cccnc2)C)C(C)C1 C1(CNC(c2c(C)cc[nH]c2=N)=O)CC2CCC1N(C(=O)CC1(C3CC3)CC1)C2 Cc1ccc(C(=O)NC2CC(C(F)C(=O)NCCc3ccc(O)nc3)C2)nn1 C1(C(=O)NCC2(C(=O)NCCn3ccnc3)CC2)CCCC2CCCN12 Cc1cncc(C)c1C(=O)NC1CC(NC(c2cc(C(F)F)no2)=O)C1 N1(C(C2CSCC(=O)N2)=O)CCOCC(F)(CNC(C2(CO)COC2)=O)C1 C1(C(N(CCCOCCN(C)C(c2sccc2Cl)=O)C)=O)C2CCC(=O)C12 C1(CC(=O)NCCC2C(C(=O)OC)C2)CCN(C(c2cnc(Cl)s2)=O)C1 c1(CN(C(CC)C)C(c2cccs2)C2CC2)ccc(Sc2ccc(Br)cc2)cc1C c1(C(N2CCC(c3ccnn3C)CC2)C(=O)NCC=C)cc(C)c(OC)c(C)c1 C(=O)(CCN(OC)C(=O)C(C)N1CCOC1=O)N(CC(CCC)O)C c1(C(N2CCC3(C(NC(=O)CC4CC(F)C4)C3)CC2)=O)c[nH]c2ncnc(O)c12 C1(CNC(C(C)(C)O)=O)CC2(CCN(C(=O)Cc3cccc(Cl)c3)C2)CO1 C(=O)(C(C(=O)NCCOC1CCN(C(=O)CCC(C)C)C1)OC)OCC N1(C(CCC#C)=O)CC2CN(C(=O)Cc3nncn3C(C)C)CC2(C)C1 C12CC(CC1O)C(=O)N2.C=CC1(C(N2CCC2C(=O)OC)=O)CCC1 c1(OC)c(O)cc(C(=O)NCC2CCC2NC(=O)CC(C)(C)C2CC2)cc1C#N Cc1cc(C(=O)NCC(C(C)C)NC(c2ccco2)=O)cnc1C(F)(F)F C1(NC(C2CC(C)CN(C(C3CCCN3C)=O)C2)=O)C(=O)OC2CCCC12 CC(C(C)C(=O)NC1CCN(C(C2CCc3nnnn3C2)=O)C1(C)C)S(C)(=O)=O c1(C(N2CCC(O)(C(N3CCC4(CC3)COC4)=O)C2)=O)n[nH]c2c1CS(=O)(=O)C2 CC1OC2CCC1(C(N1CCC(O)(CNC(=O)CN3C(=O)CNC3=O)C1)=O)C2 C1(CC(=O)N(C(C)C(=O)NC2CCN(C)CC2)C2CC2)CCC(C)(C)O1 C1(N(C)C(c2ccccc2Br)=O)CC12CCCOC2 CC1Oc2ccc(C(=O)N(C)CC3CN(C(c4cc(=O)cc[nH]4)=O)C3)cc2C1C CC1(C)CN(C(C23CCCC2CN(C(=O)CC2CCOCC2)C3)=O)CC(C)(C)O1 c1(NC(=O)OC)cc(Br)ccc1C(=O)NCC(C)(C)N(C)C Cc1nc(C)c(C(=O)NCCCOCC(=O)Nc2cccnc2)o1 Cc1[nH]c(C(=O)N(CC(C)CNC(=O)CCN2CCOCC2)C)c(C)c1[N+](=O)[O-] c1(CNC(C2CC(N(C(c3c(OC)csc3)=O)C)C2)=O)ccc(OC)nc1 Cc1oc(C(C)C)cc1C(=O)NC1CC(C)(NC(=O)CNC(=O)C(F)(F)F)C1 C(=O)(CC(C)(C)O)NCCN(C(=O)CN1CCCCC1)C CC1(C(=O)NCc2ccsc2C(=O)NCc2nn[nH]n2)CC=CCC1 c1(N2CCCC(CNC(CSC)=O)C2C)ncnc2cccnc12.C(C=O)NC Cc1cc(N2CCCC(N3CCOC3=O)C2)ncc1Br n1(CC(=O)NCC(C)NC(=O)CC2CCCCO2)c(S)nc2ccccc2c1=O Cn1c(=O)sc2cc(C(N3CC(=O)CC3C(=O)O)=O)ccc12 n1(C(C)C(N2CC(F)CC2CNC(C2CN(C)C2)=O)=O)cc2c(n1)CCCC2 Cc1cccc(C(=O)NCCN(C)C(c2cccnc2SC(C)C)=O)c1 c1(C(N2C(C(C)C)(C(=O)NCCCS(C)(=O)=O)CCC2)=O)ccc(C#N)n1C c1(C(C)(C)C)cncc(C(=O)NCCCNC(=O)CCC2CCC(=O)N2)c1 N1(C(C2(SC)CC2)=O)C2CCC1C(F)C(NC(c1cc3c(=O)[nH]ccn3c1)=O)C2 N#Cc1ccc(CN2CCN(C(=O)Cc3ccc(F)c(F)c3)C(CC#N)C2)nc1 c1(C(C(=O)NC(CCNC(C=C(C)C)=O)C)C2CCCC2)ccncc1 c1(C(=O)NC(CCC(=O)NC2(c3onc(C)n3)CC2)C)cnc2n1CCC2 OC1CC(NCC2CC2C(F)F)C1 c1(C(=O)NCC2CCN(C(C(C(=C)C)(C)O)=O)C2)nc2n(c1Cl)CCCC2 C1(C(=O)NC(C2CN(C(c3cc(Cl)ccc3Cl)=O)C2)C)C2CCC(F)(F)C12 c1(OC)ccc2c(c1)CCC2C(=O)N1CCC(NC(=O)COc2ccon2)C1 c1(CN(C(=O)C(n2nccc2C)C)CCNC(C=CC)=O)ncn(C)n1 c1(OC)ccc(SC)cc1.C(CC(C)(C)C)N(CCCON)C(=O)C=C(C)C(F)F C12(NC(CC(C)N3CCCC3=O)=O)CC1CN(C(=O)C(F)=CCCF)C2 c1(C(=O)NC(c2nocc2C(=O)NC2(C)CC2CO)C)c[nH]c2cccc(F)c12 C(C(C)(C)C#CC(=O)NC(C(C)C)c1nc[nH]n1)NC(C(C)OCC=C)=O Cc1ccc(C(=O)N(C2CC(NC(=O)C(F)(F)c3cscn3)C2)C)c2c1CCC2 C(=O)(C(C(=O)NCc1nccn1C1CC1)OC)OCC.C12(CC1)C(=O)N2 N1(C(c2c(OC)cncn2)=O)CC(CNC(=O)CC2CC(C)=NO2)CC1(C)C Cc1coc2ccc(C(N3CCC(NC(C4CCC5CC45)=O)C(O)C3)=O)cc12 C(CNC(C1CC12CC2)=O)(CC(=O)N=c1cc(C)n(C)[nH]1)OC c1(C(N(C2CN(C(C3CC3CF)=O)CC2(C)C)C)=O)ccc2ocnc2n1 c1(CN(CC(N2CCN(C)CC2)C)C)ncnc2sc3c(c12)CCCC3 Cc1nc(C(N2CC(CF)(NC(=O)CC3OCCOC3(C)C)C2)=O)cn(C)c1=O C1(NC(N2CCCCC2c2ccccc2)=O)CCC([N+](=O)[O-])CC1 C1(C(=O)OCC(C2CCC(F)(F)CC2)=O)COc2cc(Cl)ccc2C1 N1(C(C=CCOC)=O)CC2(C1)SCCC2NC(=O)CN(C(c1cscn1)=O)CC O=C(C1Cc2ccc(Cl)cc21)NCC1CC2CCC1N2C(=O)C(Cl)=CCl C(=O)(CCCC(=O)NC(C)CN(C(C1CCCC(=O)N1)=O)CC)NCCC C1(NC(C(=Cc2ccccn2)C)=O)CCN(C(C2CCOCC2)=O)CC1CO Cc1cc(C(=O)NC2CCCCCC2NC(=O)C=Cc2cn[nH]c2)cc(N)c1 c1(C(N2CC(O)(CCNC(C(CN(C)C)O)=O)C2)=O)cnccc1Br Cc1cccn2nc(C(N3CCC(OCCNC(C4OCC4(C)C)=O)C3)=O)cc12 Cc1ccccc1C(C)CC(=O)NCC(C(C)C)NC(=O)C=CCN1CCCC1 C1(NC(c2ccc(OC)nc2)=O)CC12CCN(C(=O)CCc1ccnn1C)CC2 N1(C(CC(C)NC(C2CCCSC2)=O)=O)CC(S(C)=O)C1 C12(NC(Cn3nc(C)c(Br)c3)=O)CCC1CN(C(C1CC13CCC3)=O)C2 C(=O)(C(C)(C)C(F)F)N(CC(C)CNC(c1cc(-c2ccncc2)nn1C)=O)C C(=O)(CC(C)CN(C)C)NC(C1CCN(C(C2CC(=C3CC3)C2)=O)C1)C C1(CNC(CC(CC)C2CC2)=O)CC2(CCC2)CN1C(c1ccc(N)cn1)=O c1(CN(C(=O)CC2CC3CCC23)C)ccn(CC(F)F)n1 c1(CC)ccc(C(N2CCC(CNC(=O)C=C(C)Cl)C(C)C2)=O)c(Br)c1 C#Cc1ccc(Cl)c(C(=O)NCC2CCN2C(=O)C(c2cc(F)ccc2F)=O)c1 c1(C(=O)NCC2(CNC(C3CC(OC)C3)=O)CC23CCC3)cnn(C)c1N c1(C(C)C)ccccc1C(=O)NCC1CN(C(=O)CSc2nnnn2C)C2CC12 N1(C(c2cccnc2C2CC2)=O)CCCC(O)(CNC(C2CC(C(F)F)C2)=O)C1 c1(CC)occc1C(=O)NC(C)CCNC(=O)CN(C1CCCC1)C C1(Nc2nc(N3CC(CO)CC(C)C3)c3c(n2)CSC3)COC2(CCOCC2)C1 c1(C(N2CC3C(NC(=O)C4=C(Cl)CC4)(C3)C2)=O)cc2ccccc2nc1O CC(=NO)C1CC(C(N2CC3CC2CCC3NC(=O)CCS(C)(=O)=O)=O)C1(C)C N1(c2ncnc(NCCn3c(C)nnc3)c2C)CCCC2(C=CCO2)C1 Cn1cc(NC(=O)CCN(C(c2cccc(CC#N)c2)=O)C2CC2)c(O)n1 Cn1ccc2cc(C(N3CCN(C(C4(C5CC5)CC4)=O)C(C#N)C3)=O)ccc12 N1(C(C2CC(C)C2)=O)CCCCC1CCNC(c1ncncc1N)=O N1(C(CC(C)(C)OC)=O)CCC2CCN(C(c3cc(C)nc(O)c3)=O)CC12 C1(C(=O)NC2C3CN(C(=O)CC4C=CCCC4)CC23)CCC([N+](=O)[O-])CC1 c1(C(=O)NCC(C)CNC(=O)C(C)(C)CF)cn(CCO)c(=O)nc1O CCCCCN(CCC(=O)C(CCC)SC(CNC(=O)CSC(F)F)(C)N)CCC CN1CCCC(O)(CC(=O)N(C)CCC2CCN(C(c3csc(Cl)c3)=O)CC2)C1 CC1(NC(=O)Cn2ccnn2)CCN(C(C2(N3CCOCC3=O)CC2)=O)C1 O=[N+]([O-])c1cnn2ccc(-c3ccc(Cl)cc3)nc12 C(=O)(CC(C)C(C)(C)CC)NCCN(CCC)C(c1cnn(C)c1Cl)=O c1(C(=O)N)n[nH]cc1[N+](=O)[O-].O(NC(=O)CN(C)CC)CCO C1(C(=O)OC(C)(C)C)CN(S(=O)(=O)CC2CC(C3(C=C)CCC3)C2)CCC1NC c1(N)ccc(F)cc1C(F)(F)F.c1(CNC(CCOC)=O)nnnn1C1CC1 C1(CNC(CC=CC(C)(C)C)=O)CCC(NC(C2CCC2n2ccnc2)=O)CC1 c1(-c2ccc(OCC)cc2)csc(=NCCC(=O)NC2CCOC2)[nH]1 C1(C(=O)NCc2nncs2)(NC(C2ON=C(C)C2)=O)CCc2cc(Br)ccc2C1 c1(C(=O)NCC2N(C(CC3CCC(=O)C3)=O)CC(F)C2)cccc2sncc12 N1(c2cc(NCc3ccc(Br)o3)nc(C(C)C)n2)CCC2(CCCCC2)CC1 C1(NC(C2(C(C)C)CCC2)=O)CN(c2ncns2)C2CCCCC12 c1(CCC(=O)NC23CC2CN(C(=O)CCn2ccccc2=O)C3)cccc(Cl)c1 C1(Cl)(C(=O)OC)CC12CCN(S(=O)(=O)c1ccc(C(F)(F)C(F)(F)F)cc1)CC2 Cn1nccc1C(=O)NCC(O)CNC(c1ccc(C(F)(F)F)s1)=O c1(C(N(C(CNC(C(C)=CC)=O)C)CC)=O)cc(F)cc(F)c1N NC1CC2(CC(NC(=O)C(=O)NCc3cnn(-c4nccs4)c3)C2)C1 C(=O)(CCC(C)O)NC1CC(CNC(c2c(CCC)[nH]cc2)=O)C1 N1(C(c2cnc(OC)nc2)=O)CCN(C(C2(F)CCOC2)=O)CC(O)C1 c1(C(=O)NC2C(C)CN(C(c3cc4ccsc4s3)=O)C2)ccc2c(n1)COCC2 CC1CC(C(=O)NCCCCCCNC(=O)Cc2ccccc2C(F)(F)F)=NO1 Cc1cn(-c2ccccc2)nc1C(=O)NCC1(F)CN(C(C2(CF)CC2)=O)C1 N1(C(C(C(C)C)c2cccnc2)=O)CCCC(NC(=O)C(O)C2CC2)C1C S(=O)(=O)(c1ccc(OC)cc1)N.c1(NC2CN(CCOC)C2)cc(O)ncn1 c1(C(N(C)CC2CCCN(C(C34CC(C)(CO3)C4)=O)C2)=O)ccc2c(c1)CCC2 c1(NC(c2csc(C(=O)NCCN3CCSCC3)n2)=O)cc(Cl)cc(Br)n1 CCS(=O)(=O)c1cccc(C(=O)NC2(C)CCC(NC(=O)CCCOC)CC2)c1 c1(C(N(CC(=O)NC2CCCN(C(C)=O)C2)C)=O)nnc(Cl)cc1N C1=CC2CC1C1CCC(Nc3nc4ccc(NC5CN(CC)C5)nc4[nH]3)C21 N1(C(C2C(CC(C)C)C2)=O)CCC(C)(C)C(C(=O)N(CC(C)O)C2CC2)C1 C1(C(N2C(CN(C(=O)CCc3nncs3)CC)CCCC2)=O)CC(=O)NC(=O)C1 N1(C(c2n(C(C)C)ncc2)=O)CC(NC(=O)CCc2ccco2)CCC1C CN1CCCCCC1C(N1CC(N(C)C(c2ccc(O)c(Cl)n2)=O)C1)=O c1(C(CN2CCN(C(C(C)NCCC)=O)CC2)C)ccc(Cl)cc1 c1(C(N2C(C)CC(NC(C(C)O)=O)C2)=O)cc(N)cc([N+](=O)[O-])c1 N1(C(C(C)NC(C)=O)=O)CCC2CCC12n1c(=O)ccc(NC(=O)OC(C)(C)C)c1 N1(C(CC(CC)C2CCC2)=O)CCCC(C(=O)NC2COCCC2OC)CC1 CC1CCN(C(=O)CC(C(F)F)NC(=O)C=CCN(C)C)CCS1 C1(NC(c2cc(F)cc(Cl)c2)=O)CC2CN(C(c3cc(O)cc(Br)c3)=O)CC2C1 CCC(CC(=O)NC1CN(C(c2ccn(C3CC3)n2)=O)CC(C)(C)C1)C(C)(C)C CCC(CCOC)C(=O)N1CC(N2CCN(CCCCCO)CC2)(CO)C1 c1(C(N(CCC(C)NC(C(C2CCCC2)OC)=O)C)=O)cncc(C)n1 N1(C(C)=O)CCC(C=NC(c2ccc(OC34CC3Cc3c[nH]nc34)cc2)=O)CC1 C(=O)(CC(C)(C)CNC(c1ncccc1N)=O)N(C(CC(CC)C)C)C Cc1cc(F)ccc1CN(C)CCN(C)C(C1CCCN(C2CCC2)C1)=O C(=O)(CC(C)(F)F)NCCN(CC(C)O)C(c1cnn(C2CC2)c1Cl)=O C1(CNC(c2cccnc2CNC(C2CCC(O)C2)=O)=O)CC2C=CC1C2 C1(CNC(C(C)C2CCC2)=O)C(C(=O)N(CC(O)CN(C)C)C)C1(C)C N1(C(c2cc(C)no2)=O)CCOC(CNC(=O)Cc2nnnn2CC(F)(F)F)C1 c1(C(=O)NCC(CC)NC(=O)Cc2ccncc2Cl)cncc(F)c1 CC1CN(C(C2(CC#N)COC2)=O)CC1CNC(c1ccnn1C1CC1)=O C1(=O)C(C)(C)CCCNC(=O)CC2CCCC12.N1(CCOC)CC(NC(C)=O)C1 C1(C(=O)NC(CC)CNC(=O)Cc2ccsc2)CCCN1S(C)(=O)=O CCC(C#N)(CC)C(=O)NC1CCCCC1N(C(=O)C(C(C)C)NS(N)(=O)=O)C C1(C)(C(N(C2CN(C(c3cc(N)cc(O)c3)=O)CC2O)C)=O)CCN(C)C1=O c1(OCC(=O)NCCC2CCN(C(=O)CCc3cncnc3)C2)cccc(F)c1 C1(C(=O)NCC(CN(C)C(c2cn(CCCF)nn2)=O)O)CN(C)CC1O C(=O)(CC(O)CC(C)(C)C)C(CC)CC.C12CCN(C1)CCSCCNC(=O)C2 c1(C(=O)NCC2C(C(=O)NC(c3ccsc3)(C)C)CC2)cc(O)nc(O)n1 Cc1ccc(CC(=O)NCC2(C(C)(C)O)CN(C(=O)CC3CC3)C2)cn1 C12(C(=O)OC)CCNCC1CN(S(=O)(=O)c1ccn(CCC(=O)OCC)n1)C2 c1(C(=O)NC2C(NC(CSC)=O)CC2)cc(CCN2CCCCC2)on1 N1(C(c2c(CC)nco2)=O)CC(C(=O)NC2CCCC2CN(C)C)C2(CC2)C1 c1(C(C(=O)NCCNC(c2cc(Cl)n[nH]2)=O)OC)cc(F)cc(F)c1 c1(C(C(=O)N(CCNC(c2ccns2)=O)CC)=O)c(C)[nH]c2ccccc12 c1(C(=O)NCC(CCOC)NC(=O)C2=CCCC2(C)C)cccc2cccnc12 C1(CC(=O)NC2CC(C)SCC2)CC2(C1)CN(C(C13CCC(CC1)C3)=O)C2 CC(C)(C)CCC(=O)NC1CN(C(C2(c3ncco3)CC2)=O)CCC1C(F)(F)F c1(C(=O)NCC2C(NC(C3CC=C(C)CC3)=O)C2)c[nH]c2cccc(N)c12 c1(NC(c2c(C)noc2C)C)cc(Br)ccc1[N+](=O)[O-] C1(N(C(C)CC(=O)OC)C(=O)COCC(C)(C)C)CCCCCC1 C(=O)(CC(O)CC(C)C)NC(c1ccc(C)cc1)CNC(C(C=CCCC)O)=O C1(CNC(C(C)NC(N)=O)=O)CC2CC(C1)N(C(c1ccco1)=O)C2 N1(C(C(CC=C)(F)F)=O)CCCC(F)(CNC(=O)CCC2CCC(=O)NC2)CC1 C12CN(CC1C)C2=O.CCC(CN1CCC(C(=O)NC(C)(C)C)C1)CC c1(OC)cc(C(=O)NC2CN(C(c3ccc(F)c(Br)c3)=O)C3CC23)cc(OC)n1 CC12CCCN(C1)C2.c1(NC(c2cnc(-c3ccccc3)s2)=O)cc(F)c(Cl)cn1 CCCCC(CCC)NC(c1conc1CC)=O CC(C)CC(F)(F)C(=O)NCC1CN(C(=O)CN2CCC(C)(O)C2)CCC1(C)C C1(CCN)CCC(=O)CC1.n1(NC(CN(C2CCSC2)C)=O)ccnc1 C=CCCC(C(=O)N1CCCC(CCC)C1)NC(C1CC1C(F)F)=O C12(CCNC(CCC3(C)CC3)=O)CCC(C1)N(C(c1cccc(F)c1N)=O)C2 C(=O)(C(CO)C(C)(C)C)N(CC(CNC(C1(C(C)O)CC1)=O)(C)C)C c1(OC)cc(C)cc(C(N2CCN(C(=O)Cn3cnnc3O)CC(O)C2)=O)c1C O=S(=O)(c1ccc(NCC2CCC2CO)cc1Br)NC1CCOC1 C1(C(N2C(C(=O)NCC(C3CCCCC3)C)C(C)C2)=O)CC2CC(=O)C1O2 c1(CNCC2N(Cc3cccc(C(=O)O)c3)CCOC2)cc(Cl)ccc1Br Cc1[nH]nc2c(C(N3CC(NC(c4cc(Cl)c(Cl)cc4O)=O)C3)=O)cccc12 C1(NC(c2ccc(C=C)cc2)=O)CC2CCC(C1F)N2C(=O)CC1(C)CCCO1 C1(C)(C(c2n(C(CC)(C)C)nnn2)NCC(CC2CC2)CO)CCCCC1 c1(CN2CCC(CC(=O)Nc3cccc(Cl)c3F)C(O)C2)cc(Br)c(F)cc1Cl c1(OC)c(C(N2CCCC(NC(C3CCCOC3C)=O)CC2)=O)cc(F)cc1F c1(C(=O)NCCOC2CN(C(c3n(C=C)ncc3)=O)C2)cc(Br)c(O)nc1C c1(CCC(=O)NCCN(C2CCCCCC2)C(c2cc[nH]n2)=O)cncc(F)c1 CC1(C)Cc2n[nH]cc2CN(S(=O)(=O)c2cccnc2)C1 C1(OC)CC2(CCC(C(=O)NC(C3CCN(C(=O)OC(C)(C)C)C3)C)CC2)C1 N1(C(CCCNC(C)=O)=O)CCCCC(NC(=O)CC2CC3(CC3)C2)C1 c1(C(=O)NCC23N(C(CC(C)CF)=O)CC(C2)C3)nn(C)c2ccc(F)cc12 C1(NC(C2CCOC2=O)=O)COC2(C1)CN(C(=O)Cc1ccsc1Cl)C2 Cc1cccc2c(C(N3CCN(C(=O)CC4(CO)CCCC4)C(C)C3)=O)c[nH]c12 CCCC(C(=O)NC)NC(C1CN(C(=O)CC(C)n2cccn2)CCO1)=O C(=O)(C#CC1CCOCC1)OCC.CCC(C)CC1C(=O)c2ccc1c(OC)c2 c1(C(=O)NC(C)CCNC(=O)CN2CCCNC2=O)ccc(Br)c(F)c1 N1(C(c2c(C)n(C)cc2)=O)CCOCCC1C(=O)NC(C)Cc1ccco1 c1(C(=O)NC2(CNC(c3ccn(C)c3)=O)C(C)CCCC2)cccn2cnnc12 c1(C(=O)NC2(CCNC(=O)CC3CC(F)(F)C3)CCC2)csc([N+](=O)[O-])c1 c1(CC)cccc(C(=O)NCC(CNC(=O)CCNC(=O)COC)CO)c1F C#Cc1ccc(C(=O)NC(C2CN(C(c3cnc(C)c(C)c3)=O)C2)C)c(OC)c1 N1(C(C(CC)(CC)CO)=O)CC(CNC(=O)CCc2nc[nH]n2)OC2(CCC2)C1 N=c1[nH]c(CO)ncc1Br.n1(CC(N2CC(OCCOC)C2)=O)cc(C)nn1 C(=O)(C(C)(C)C(C)(F)F)NCC1(OC)CCN(C(c2ncc(F)cc2F)=O)C1 c12[nH]c(C)c(OC)c1C(=O)NCC2.C1(SC)CCCC1CF.C1C(=O)O1 C(=O)(C(C)(COC)CC)NC(C1(O)CCN(C(CN(CCOC)C)=O)C1)C c1(OC)ncc(C(=O)NCCC(O)C(=O)NC(C)(C)C(C)(C)O)cn1 C1(NC(COC2CN(C(c3nc(OCC)oc3)=O)C2)=O)CCOC(C)C1 N1(C(C2=C(C#N)CCC2)=O)CCC2(CCCN2C(=O)CCC(N)=O)C1 N1(C(CCOCCNC(Cc2cccc(C#C)c2)=O)=O)CCN(C)C(=O)C1C C1(NC(Cc2cccc(C)c2F)=O)CN(C(c2ccnn(C)c2=O)=O)C2(CCC2)C1 C1(CNC(Cn2c(C)cnc2)=O)CC2COCC2N1C(C1(CF)CC(=O)C1)=O C=C(C)C(C)(C)C(=O)N1CC(C(O)C(=O)N(C2CCN(OC)CC2)C)C1 c1(C(N(C)CC2N(C(CNC(C(CC)C)=O)=O)CC(F)C2)=O)nc(C)n(C)c1C C1(NC(c2cc[nH]n2)=O)CN(C(c2cc3n(n2)CCC3)=O)C2CCCC12 C1(NC(c2ccncc2C(F)(F)F)=O)CN(C(c2nc(Cl)c(Br)s2)=O)CC1(F)F C1(OC(C)=O)C=CC(NC(=O)CC2(C)CN(C(c3ccc(ON(C)C)s3)=O)C2)C1 c1(NC=O)ccnc(C(C)C)c1.c1(CC)cc(C(=O)N(CCC(=O)NC)C2CC2)on1 C1(COC)CC2(CCN2C(=O)CCCN(C(=O)CCC2CC2(F)F)C)C1 C1(c2cc(OC)c(CC(C)C)c(OC)c2)NC(=O)N(C2CC2)C2=C1C(=O)NC2C C(C(C)(C)CC(F)F)NC(C(n1cc(-c2cccc(COCC)c2)nn1)C)=O C1(CNC(c2conc2C2CC2)=O)CCCCN1C(=O)CN1CCCNC1=O N1(C(C2(COC)CN(C(C(C)SCC)=O)C2)=O)CC2CC(CO)C(C2)C1 C1(C(N(CCCNC(c2ccn3ccsc23)=O)C2CC2)=O)CC2(C1)CC21CC1 N1(C(c2ccc(OCC)cc2)=O)Cc2sccc2CCC12CCC2 C1(CC(=O)N(CC(CCC)C)C)CC(C)N(C(c2cn(C)nc2C)=O)C1 N12CCOCC1CC2=O.C1(NC(CCC#C)=O)CCOC1N.C(C)C c1(C(=O)NC2CN(C(C3C(CC)CCC3)=O)C2)cc2cccc(C)n2n1 N1(C(c2c(CCC)nco2)=O)CCOC(CCC(=O)NC(COC)CCO)C1 CN1CCC2(CCN2C(=O)CC2CCCN(C(C3(O)CCSCC3)=O)C2)C1 N1(CC(N2C(CCSC)CCC2)=O)CCC(c2cn[nH]c2)CC1 CC1CN(C(C2COC(CNC(C34CC(C)(CCO3)C4)=O)C2)=O)CC1(C)CO c1(C(=O)NCc2cccc(OC)n2)ccc(C)c(OC2(C(=O)OC)CCC2)c1 c1(C(CO)NCC2(NC(c3cc(C)c(Br)s3)=O)CC2)ccc2c(c1)OCO2 N1(CC)CCCC2C(C(=O)O)C(C)(C)C12.c12cccc(n1)C(=O)N2 N1(C(Cc2c(C)n[nH]c2C)=O)CCN(C(=O)C(C)(F)C(F)(F)F)CCC1C C1(S(N)(=O)=O)(C(=O)NC(C)C(CO)NC(=O)COCCF)CC1 C1(NC(c2cc(C)[nH]n2)=O)CC2CCC1CN2C(=O)CC1C=CCCC1 CC1CCCCCC1NC(=O)CCCCNC(=O)CC1CCN(C)C1=O c1(N2CCC(C(C)C(=O)NC(C)C)CC2)ncnc2c1nnn2Cc1cccs1 c1(C(=O)NC(CNC(c2c(C)csc2)=O)C(C)C)cccn2nnnc12 c1(C(=O)NCCSC)ncccc1-c1cn(CC(C)NC(CC(C)SC)=O)nn1 n1(CCCOC(C)C)nnc2ccccc2c1=O.C12CCOC1CNC(=O)N2 C1(NC(C(CC)SC)=O)CCN(C(=O)Cn2ncnn2)C12CCC2 CCC(C)CC(C)C(=O)NCC1(C(N2CC(c3nncn3C)C2)=O)CC2(CC2)C1 C1(C(C)NC(=O)COCc2nc[nH]n2)CCCCN1C(c1sc(SC)cc1C)=O c1(OC)ncc(C(=O)NC2CCCC2CC(=O)NCCC(C)C)cn1 c1(C(N2CC(NC(C(CC)C(C)C)=O)C2)=O)oc([N+](=O)[O-])cc1C C(CC(C)C(=O)NCc1ccc(CN2CCCCCC2)cc1)=CCC O=S(=O)(c1cc(F)ccc1F)Nc1cccc2ccccc12 Cc1cn2c(C(N3CCN(C(c4cnnc(O)c4)=O)C(C(C)C)C3)=O)cnc2s1 c1(CC)cc(C(N2CCN(C(=O)C(F)=CCCF)C(C3CC3)C2)=O)ccc1F c1(C(=O)NC2CC(NC(c3c(C)cc(Br)c(F)c3)=O)C2)ccnc2ccccc12 C1(NC(c2ccc(C)nc2)=O)CN(C(c2occc2C)=O)CC2(CC2)C1 C(=O)(CCC(CF)CF)N1CC2C(CC(=O)NC(C)(CO)C3CC3)C2C1 C1(C(=O)NC2(C)CC(NC(CCc3cc(C)on3)=O)C2)CC2CCC(C1)N2C C(=O)(C1=C(C)CCCC1)NCCC1CCN(C(C2CN(CC)C(=O)C2)=O)C1 c1(C(N2CC(C)C(NC(=O)CN(CC(C)(C)C)C)C2)=O)cc(C#N)ccc1N C=C=CCCC(=O)N1C(C(=O)NC(C)COC(C)=O)C2CCC12.OCC C1(=O)CCCC(=O)N(C2CC2)CC(=O)N1.N1(CC)CC(C)SC(C)C1 c1(-c2n(Cc3ccc(O)cc3)nc(COc3ccccc3)n2)c(Cl)cccc1Cl C1(C(=O)NCC(CO)NC(C=Cc2n(C)cnc2)=O)CCc2cnn(C)c2C1 c1(C(=O)NCC(C)(C)NC(=O)C(O)C2CCCC2)ccc(Cn2cccn2)cc1 CCCCCC(O)CC(=O)NCC(C)(F)CNC(=O)C(C)=C1CC1 Cc1nccc(C(=O)NC(Cc2ccoc2)C(=O)NCC2(CO)CCC2)c1N CC(C)C(C)(CNC(=O)Cc1cccnc1C(F)(F)F)NC(=O)CC(F)F CC1CCC(c2nnnn2-c2ccccc2)(NC(c2ncc(Br)s2)C2CC2)C1 CC1CC(C(N2CC(C3CC3)(CO)C2)=O)CN(C(c2ccn(C)n2)=O)C1 CCCCC(F)(F)C(=O)NC1CC(C(F)C(=O)NCCCC2CCC2)C1 O=S(=O)(c1c(F)cc(Cl)cc1F)NC(CC(F)(F)F)c1ccc(Br)cc1 C1(NC(CNC(N)=O)=O)CCCC1(C)CNC(c1csc(-c2ccsc2)n1)=O c1(NC(C2C(c3c(C)ccs3)C2)C)ccc(S(=O)(=O)NCc2nccnc2C)cn1 c1(C(=O)NC(CNC(C2CCC(SCC)CC2)=O)C(C)C)cc(OC)cc(C)n1 C#CCC(CC(F)F)C(=O)N1CC(O)(CCNC(=O)COc2cccc(C)c2)C1 N1(C(c2n(C)ccc(=O)c2)=O)CCCC(C2CN(C(=O)C3CC3)C2)C1 CN1CCN(C(=O)C=Cc2cccnc2)C(CNC(C2CCCS2(=O)=O)=O)C1 Cn1ccc(C(c2nnnn2C(C)(C)C)NCC2(c3ccccc3)CCCO2)n1 N1(C(c2c(CC)occ2)=O)CC(NC(c2ccnc(F)c2OC)=O)CC12CCC2 CC(C)(C(=O)NCCCCCCO)C1=CCN(C(=O)Cc2cccs2)C1 N1(C(C(C)=C2CC2)=O)CCCC(Nc2ncnc(C)c2F)CC1 C#CCCCCCC(=O)NC1(C2CCN(C(=O)C3=C(C)CCCC3)C2)CC1 c1(C(N(C(CNC(C(C)Oc2ccccc2)=O)C)C)=O)cc(Cl)ncc1F c1(OC(C)C)ncc(C(=O)NCC2CCC(NC(c3ccns3)=O)CC2)cc1Cl C1(C(=O)NCCN2CCN(C(C(C)CCO)=O)CC2)CNC(=O)CC12CCOC2 Cn1cc(C(=O)NC(CC(N)=O)c2ccccc2)c(=O)c(Br)c1 c1(NC(C2C3CN(C(C4(C)CCC4)=O)C2C3)=O)cc(C#N)c(F)cc1Br c1(NC(C2CCN(C(c3ccncc3Br)=O)CC2O)=O)ccc(Cl)c(I)c1 c1(NC(=O)NCCOC)nc2cc(OC)ccc2o1.C1(OC)CC(OCC)C(O)C1OC N1(C(c2cn(CCNC(c3cn(C)nc3)=O)nn2)=O)CCOCC(CO)C1 C1(C)(CNC(c2c(CC)nns2)=O)CN(c2cc(Cl)ncn2)CCO1 c1(CSCC)cccc(C(=O)NC(C)CCNC(=O)C(C)(C)c2ccno2)c1 C1(CNCc2ccc(SC)cc2)CC(C)CCN1C(=O)C(CO)c1ccccc1 C1(C(N(CC(C)O)CCNC(c2ncn(C)n2)=O)=O)CCC2(CCCC2)C1 c1(SCC)nccnc1C(=O)NC(C)CCN(C(=O)C(C)N1CCC1)C CN=c1nc(N2CCCC(CNC(C)=O)C2)[nH]c(=NC2CCOC(C)(C)C2)[nH]1 N1(C(c2c(OC)n[nH]c2)=O)CCCCC(NC(C2CC=CCC2C(F)(F)F)=O)C1 CCCC(C)(O)CNC(c1cnn(CCNC(=O)CNC=O)c1)=O C(=O)(C1CCc2cccnc21)NC(C1CN(C(c2cscc2C#N)=O)CCO1)C N1(C(C2CCCS2)=O)CCC(NC2CN(C(C3CC3[N+](=O)[O-])=O)C2)CC1 C1(COC)CN(C(c2cc(C)ccc2O)=O)CCN1C(c1ncnc(C)c1C)=O Cc1nc2cc(C(=O)NC3(CO)CCN(C(C4CCC(C)C4)=O)CC3)ccc2o1 C1(CNC(c2ccc(CCC)cc2)=O)CC(F)(F)CN1C(c1cc(OC)ns1)=O C1(NC(Cc2n(C)ncc2)=O)CCN(C(=O)C(C)(C)C2CCOC2)CC1F C1(C(=O)NCC(=C)Cl)CCCCN1C(=O)Cc1n[nH]c(C)n1 C=CCC(CC=C)C(=O)N1CC2(CCC2)CC1CNC(=O)Cc1cscn1 CC1(C(=O)N(CC(=O)NCCN=S(C)(C)=O)C2CC2)CCC(O)CC1 CCC(Cc1ccccc1)CC(=O)N(CCCNC(=O)C(F)C(C)(C)O)C1CC1 C(c1ccc(Cl)c(C(F)(F)F)c1)=CC(=O)NCC(CC)NC(C12CC(CO1)C2)=O c1(C(=O)NC2C(NC(=O)CCC=Cc3ccccc3)C2)cccc2[nH]cc(Cl)c12 C1(NC(C2C(CC)CCN2C(=O)C(C)=C2CCC2)=O)CCCN(C)C1 C(=O)(C(O)CC(F)F)NCC(CNC(c1c(N(C(=O)OCC)C)cccc1)=O)O C=CCC(CNC(c1sccc1Cl)=O)NC(c1ccc(F)s1)=O c1(C(C(=O)NCCCC(=O)OCC)N(C)CCF)cnc(N2CCOCC2)nc1 C(C)(CN=c1[nH]c2c(c(=NCCCCCCO)[nH]1)CSC2)c1c(OC)cccc1 N1(C(c2n(C)ncc2N)=O)CCC(C2CC2)C1CNC(=O)CC12CCC(CC1)C2 N1(C(CSCC=C)=O)CC(NC(c2ccccc2-c2nnc(C)o2)=O)CCC1C N1(C(C(CC)O)=O)CC(NC(=O)C=Cc2cc[nH]n2)C(O)C1 CC(C)CC(F)C(=O)NCCN1CCN(C(=O)Cn2cc(CO)nn2)CC1 CC1(C)C=C(C(=O)N2CCC(C)(C(=O)NCc3c[nH]nc3C3CC3)C2)C1 c1(C(N2CCC(C)(NC(CCCC(=O)NC)=O)CC2)=O)cccc2c1CCO2 C1(NC(C=C(CCC)C)=O)CCCC(NC(=O)Cc2ccc(C(=O)C(C)(C)C)s2)C1 c1(C(N2CCCC(N(C(C(C(CC)O)C)=O)C)CC2)=O)cccn2nncc12 N1(C(c2cc(CNC(=O)CCc3cncs3)on2)=O)CCC(C2(C)CC2)C1 c1(C(=O)NC2(CCNC(COC(CC)C)=O)CCC2)ccncc1Cl C#CCC(C(=O)NC)NC(C1CCN(CCSCCCO)CC1)=O N1(C(c2ccc([N+](=O)[O-])c(C(F)(F)F)c2)=O)CC(C(=O)O)Cc2ccccc21 CCC(C)CC(C(=O)OC(C)(C)C)NC(=O)Nc1cccc(C(C)(C)O)c1 C1(CNC(CCCC(C)O)=O)CC2COCC2N1C(c1ccc2ccoc2c1)=O C1(C(N2C3CN(C(CC4CCC(=O)O4)=O)CC2CC3)=O)CCc2ncncc2C1 Cc1nn(C2CCCC2)c(C)c1CCC(N1CC(C2CC2)C1CO)=O N1(C(c2c(C)n(C)nc2)=O)CCC2CC2(C(=O)NCCc2nc(=N)[nH][nH]2)CC1 c1(C(N2C3C(NC(c4cc(F)ccc4F)=O)C(C3)C2)=O)coc2c1C(O)CCC2 c1(C(=O)NCC23OCC(NC(C4C(CC)OCC4)=O)(C2)C3)cc(F)c(F)c(O)c1F C1(C(N(C2CCN(C(c3coc(N(C)C)n3)=O)CC2)C)=O)CC12CC(F)(F)C2 N1(C(c2ccc(C)c(F)c2)=O)CC2CCN(C(=O)C=CC(C)(C)C)C2C1 c1(C(=O)NC(C2CCOC2)CNC(C2(Cl)CC23CCC3)=O)cc(F)cc(Cl)c1 c1(C(=O)NC(CC)CN(C(=O)C(F)C(C)C)C)cc(C)c(N)cc1F O=C(CCCC(F)(F)F)N1CC2CC(C1)N2C(C12CCCCC1OCC2)=O Cc1nc(O)ccc1C(N1CC(O)CC1(C)C(=O)NCCC1CC(=O)N(C)C1)=O c1(C(=O)NC2CC2CNC(C2(C3CC3)CC2)=O)ccc2c(c1)S(=O)(=O)NC=N2 C1(C(=O)O)(NC(=O)NC(c2c(C)nc(SC(F)(F)F)s2)C)CC(O)C1(C)C c1(C(=O)NC2CC(NC(C(C(C)C)OC)=O)C2)cnc2n1CCC2 N1(C(C(C)OC2COC2)=O)CC2(C1)CN(C(c1ccc(N)cn1)=O)C2 c1(OC)cc(CNC2CCCN(c3ncc4n3CCNC4)C2)cc(OC)c1Br N1(C(C2C(C(C)C)(OC)C2)=O)CC2(CCN(C(=O)CO)CC2)CC1C N1(C(C(C(C)C)c2ccccc2)=O)CCC(NC(c2cc(Br)c[nH]2)=O)C(F)C1 c1(CC(=O)NCCCCCNC(C(CC)F)=O)cccc(Cl)c1 c1(C(N2CCC(CNC(CCCOCCC)=O)(CO)C2)=O)c(C)oc(C)c1C C12C=CCCC1C(=O)O2.c1(CN(CCOC2COC2)CC)ccccc1 c1(CCC(N2CC(C(=O)OC)C2(C)C)=O)c(C)nn(-c2ccccc2)c1C.CC N1(CC(=O)NCC2CCCC(CNC(C(C)(C)F)=O)C2)CCC(=O)NC1=O c12cc(cnc1C)C(=O)N(CC)CCNC2=O.C(=O)(C(C)P(C)(C)=O)NC c1(OC)ccn2cc(C(=O)OCC(N3CCN(C)CC3)C(C)C)nc2c1 C1(OC(C(=O)NC(c2c(OC)ccc(OC)c2)C)=O)C(C)C(CO)C12CCC2 C1(CCC)(NC(c2cc[nH]c(=N)c2)=O)CCN(C(=O)CCCNC(C)=O)CC1 c1(C(=O)NCC2CCC(F)(CNC(CC(CC)SC)=O)C2)cc2occc2s1 c1(OC)cc(OC)nc(C(=O)NCC#CCNC(=O)CC2COCC(C)(C)O2)n1 Cn1cc(C=CC(=O)N(CCNC(=O)C(c2ccccc2F)C)CC2CC2)cn1 N1(C(C2(CNC(CC3C(C)OCC3)=O)CCCO2)=O)CC2(C)CCC2(C)C1 N1(CC(=O)NCC(c2ccc(F)cc2)NC(CSC)=O)CCS(=O)CC1 C(=O)(C#CC(C)(C)C)N(C1CCN(C(c2c(C)cc(CC3CCC3)o2)=O)C1)C C1(NC(C(C(CC)C)C)=O)CCN(C)C12CCCN(C(=O)COC(F)F)C2 Cc1ccc(C(=O)NCC(CO)NC(c2scnc2C2CC2)=O)cc1[N+](=O)[O-] CCN(OC)C(=O)CNC(C1CCCN1C(=O)CNc1ccccn1)=O CCC(C)(C)C(O)C(=O)N1CCN(C(=O)CC2(C(C)C)CC2)CC1CO c1(CC)cccc(C(N2CC(O)CC2(C)CNC(=O)C2=NNC(=O)C2)=O)c1C C1(NC(c2c(C)cncc2)=O)CC2CCC(C1)N2C(=O)C(C)Cc1ccnn1C C1(C(=O)NCC(C2CCCC2)NC(c2cn(CC)nc2)=O)(OC)CCC12CCC2 CCC(C)(CCC(C)C)C(=O)NC1CCCC2CN(C(=O)C=C(C)C3CC3)CC12 c1(C(=O)NCCOCCCO)cccc(-c2cccc(CN(C)C)c2)c1 O=C1NCC(C(=O)N2CC(F)(CNC(C3CCCS3)=O)C2)n2nccc21 C1(CC(=O)NC2C(O)CCN(C(C=C(CCN(C)C)Cl)=O)C2)CC2(CCC2)CCO1 N1(C(CC2(OC)CCC2)=O)CC(CNC(=O)CSc2cccc(F)c2)CC(C)C1 c1(C(N2C(CCCC)CCC2)=O)cccnc1CNC(C1CCCC(O)C1)=O C=CCC(C)(C)C(=O)NCCN1CCN(C(c2cc(C3(CC)CC3)on2)=O)CC1 CCC(C)CCCCC(=O)N1CC(O)(CNC(=O)C=Cc2ccccc2Cl)C1 c1(OC)ccc(C)cc1NC(=O)CC1COCCN1C(=O)CC1=CCCC1 C1(C(N(C(C(=O)NCC2(CC)CCC(=O)N2)C)C)=O)CCC(C2CC2)C1 CC1CCN(C(c2c[nH]c(=S)cn2)=O)C1C(=O)N(C1CCC(CO)CC1)C C1(NC(c2c(CC)occ2)=O)C2CC3C1C3C2C(=O)NC1CCCC(C)C1 CC1(C)CC(C(=O)NCc2cncs2)CCN1C(C1CCCC1C1CC1)=O c1(NC(=O)NCCCc2cccnc2C(F)(F)F)cc(F)ccc1Cl C1(CCC)C(C)CCCN1C(C1CCN(C(C2CCCSC2)=O)C1)=O Cc1c(C(N2CCCC2CN(C)C(c2cc(Br)c[nH]2)=O)=O)sc2cncn12 N1(C(Cc2c(C)cccc2C)=O)CCN(C(C23CC=CC(C2)OC3)=O)CC(O)C1 N1(C(CSCCC(C)C)=O)CCCCCC1CNC(C1CC(=O)NC(C)C1)=O C(=O)(C(F)CC(C)(C)NC(c1c[nH]c2ccncc12)=O)N1C(CC)CC1 N1(CCc2cn(C3(C(=O)O)CCCOC3)nn2)CCOCC2(C1)CC2(F)F C#CC1CN(C(=O)CC2CCSC2)CCN1C(=O)C(=Cc1cccnc1)C C1(NC(C(C)OC)=O)CC(NC(=O)COc2ccccc2F)CC1O c1(C(=O)NCCC(C)NC(c2c(C)scn2)=O)c(F)cc(Cl)cc1F c1(N2C(CNC(c3c(C)ccnc3Cl)=O)COCC2)ncnc2ccsc12 C1(C)(N(C(C)=O)CCNC(c2ncc(C)o2)=O)CC(OCc2ccccc2)C1 CCCC(C(=O)N1CC(O)(C(N(C)Cc2sncc2C)=O)C1)NC(c1ccco1)=O C1(CNC(c2ccc(C(C)=O)cc2)=O)CC12CCN(C(C1CCSC1)=O)CC2 c1(C(N2C(CNC(C3CC=CC3)=O)C=CC2)=O)ccc2cccc([N+](=O)[O-])c2n1 CCC(CC(=O)N1CC(O)(C(C)NC(C2C(C3CC3)C2(F)F)=O)C1)CC(C)C c1(OC)cnc[nH]c1=NCCC(C)NC(c1c(C2CC2)cnn1C)=O c1(C(=O)NCCCN(C(c2c(SCC)cccn2)=O)C)cc([N+](=O)[O-])ccc1O c1(NC2CN(C(=O)OC)C2)cc(C)ccc1C(=O)NC(C)=O CCC(CC(=O)NC1C2CCC(C2)C1C(=O)NCCCC(C)(C)CO)C(F)F c1(NCCOc2ccc(C)cc2)ccc(OCCCn2ccnc2)c(F)c1 C=CCC(CC(C)C)C(=O)NC1CC12CCN(C(=O)CC1CSCCO1)C2 c1(NCC2C(NC(c3scc(C)c3)=O)CCC2)ccc([N+](=O)[O-])cc1Br c1(C(N2CCCN(C(C3(C)CCC(=O)C3)=O)CC2)=O)cc2n(c1)CCOC2 C1(CN(C)C(c2cc[n+]([O-])cc2)=O)CN(C(C2CC3CC3C2)=O)CCO1 c1(C(=O)NCC2(C)CN(Cc3cc(F)cc(Cl)c3)C2)cc(I)c(F)cc1Cl CCC(C)(CNC(C1CCCN(C(=O)Cn2ccnc2)CC1)=O)C(N)=O Cc1ccc(=O)n(CC(=O)N(C2C3CN(C(C4CC(F)(CF)C4)=O)CC23)C)c1 C(CN=c1[nH]c(=NCC(C)N2CCOCC2)[nH]c2c1COC2)N(C(=O)OCC)C N1(C(CC(COC)(C)C)=O)CCC2(C=C(C(=O)NCC3CCCC(OC)C3)C2)C1 Cn1ccc2cccc(-c3c[nH]nc3C(=O)Nc3cncc(F)c3C#N)c12 C1(NC(C2N(C(C)=O)CC2)=O)CCC(CNc2cc(Cl)ncn2)CC1 Cc1c(C=CCNC(=O)NC2CN(C(C)C)CC2C(F)(F)F)cnn1C Cc1oc(C(=O)NCC23CC(CO2)N(C(c2cncc(N)n2)=O)C3)cc1[N+](=O)[O-] C(=O)(C1CCc2scnc21)N(C(C)CNC(=O)C(F)CC1CCCC1)C N1(S(=O)(=O)c2cccs2)CCN(N2CCCC2C(F)F)CC1 C(=O)(CC1CNc2ccccc21)N(C1CN(C(c2cccnc2)=O)CC12CC2)C CC(C)C(C)(O)CNC(c1c[nH]nc1CNC(C1COCCC1C)=O)=O C12(NC(c3coc(C(F)(F)F)n3)=O)CCCC1CN(C(=O)CC(F)(F)Cl)C2 N1(C(CC2C(CC)C2)=O)CC2CC(N(C(=O)CCc3ncc[nH]3)C)C1C2 CCCC(C)CC(=O)N1CC2CC(NC(=O)C(C)(C)n3ccnn3)C1C2 Cn1ccc(=NC(=O)C(F)Cl)[nH]1.C(CC(=O)O)N1CC1 C=CCCCC(=O)NC(C)CCN(C)C(c1cccnn1)=O CCCC(CCC)C(=O)NCC(c1nn[nH]n1)C.C12CCCN(C1)C(=O)C2 c1(C(=O)NC2CCN(C(C3CCCN(C)C3)=O)C2(C)C)cc2ccc(Cl)cc2[nH]1 N1(C(C2(C#C)CC2)=O)CC(N(C)C)C(NC(=O)CC2(OCC)CC2)C1 c1(NC(CC2OCCN(C(C(C)(C3CCC3)OC)=O)C2)=O)ccc(Cl)nc1C N1(C(C(=O)NCCNC(C)=O)=O)CCN(C=O)CCC12CCC2.c1(OC)cccnc1 C1(NC(c2ccc(C(C)C)s2)=O)CC12CCN(C(c1ccnnc1)=O)C2 n1(CC(=O)NC2CCN(C(c3c(C)cnn3C)=O)C23CC3)nnc2c1CCCC2 C1(C(=O)NC(C)C(c2ccccc2)NC(=O)C(N)=O)CCCCN(C)C1=O n1(CC(N2CC3(CN(C(C4C(=C)C4)=O)C3)C2)=O)ncc2ncccc12 N1(C(C(CCC)NC(N)=O)=O)CCCC(C(=O)NCCOCCCF)(CC)C1 c1(N2C(C(C)(C)NC(C3CCCOC3)=O)CCC2)ncc(Cl)cc1[N+](=O)[O-] C(C(C)(O)CCCO)NC(=O)NC1CCN(Cc2nc(C)on2)C1 Nc1cc(F)ccc1C(=O)NC1CC(CCNC(=O)CCC(F)(F)F)C1 c1(CCC(=O)NC2C(NC(CCC=CCC=C)=O)COC2)cc(C)sc1C C1(CC(=O)N(CCCNC(c2ccc(Br)o2)=O)C)CCC2(CC2)CO1 C1(NC(C23CC(NC(C(C)OCC=C)=O)(C2)C3)=O)CCn2nccc2C1 C1(C(=O)NCc2cc(C(=O)Nc3c(C)ncnc3)ncc2)CC2CCCC2C1 C1(COc2snc(C(=O)OC)n2)CCN(C(=O)CN2CCCCC2CO)CC1 Cc1cc(C(N2CCN(C(=O)C3=CCC3)C3CC23)=O)c2nc(C)n(C)c2n1 c1(C(CC(N2CCC(C)(NC(c3c(CC)non3)=O)C2)=O)C)ccc(F)cc1F Cn1ncc([N+](=O)[O-])c1NC1CCN(C(C2CCCC23CC3)=O)C1 c1(C(=O)NCC2CCN(C(C(F)OC)=O)C2(C)C)c(C)nc(C2CC2)nc1O C#CCCCCCC(=O)N1CC(NC(c2ccnc3[nH]cnc23)=O)C(C(F)F)C1 c1(OC)cccc(CCC(=O)NCC2CCC(NC(=O)CCc3cccs3)C2)c1 C1(C(=O)OC)CC2(CCCC2)CN1C(c1ccc(OC)c(Cl)c1)=O N1(C(CCc2nc(C)sc2)=O)CCC2(CCC2)C(NC(=O)C2=CCOC2)C1 C1(C)(C(c2nnnn2CC(F)F)NCCC(=O)NC(C)C)CC2(C1)OCCO2 CC(C)CCCC(C)CNC(=O)C(C)C1(O)CCC1 c1(C(=O)NCC2CN(C(c3cc(CC)c(CC)o3)=O)C2)cnn2c(C)ccnc12 c1(OC)ccc(NC(=O)CC2CCC(C)N(C(=O)CCC=CC(C)C)C2)cc1C N1(C(C(CCCC)NC(c2ncn(C)n2)=O)=O)Cc2ccncc2C1 CON(CCC(=O)N1CCCC1CC(N)=O)C(=O)CCC1CC1c1ccco1 C1(O)(C(CC)C(=O)NC(C2(O)CN(C(=O)CCOCCSC)C2)C)CCCCC1 C12(CNC(Cc3cn(CC)nc3)=O)CCC(CC1)N(C(C1CC3CCC3C1)=O)C2 c1(Nc2ncc(C(=O)OC)c(C)c2)ccc(Cl)c(Cl)c1C N1(C(C(C)C#N)=O)CCC(C)(C(=O)NC(C)Cc2nn[nH]n2)C1 Cc1ccccc1C(CNC(=O)C(C)CN(C)C)NC(=O)C(C)(C)CC1CC1 C(c1cccc(Cl)c1)=CC(=O)NC1(C)CCN(C(=O)COC2CC=CC2)C1 N1(C(C2CC(C)OCC2)=O)CCC(F)(CNC(=O)C(C)(C)F)CC1 N1(C(c2cc(C)c(C)[nH]2)=O)CC(NC(c2cc[n+]([O-])cc2)=O)CC12CCCOC2 C1(C(=O)NCC2(OC)CN(C(=O)CC(C)N3CCCC3=O)C2)CCCCC1(F)F N1(C(C(C)OC)=O)CCC2CCCN(C(=O)CC3(O)CCCC3)C2C1 C1(CCNC(Cc2n(C(C)C)cnn2)=O)CCCN(C(=O)CC2CSC2)C1 N1(c2nccc(C(C)(C)C)n2)CCC2CCN(C(C3(CN(C)C)CC3)=O)CC2C1 c1(C2C(NC(=NCc3c(C(C)C)cccc3)NCC(F)F)C2)cc(F)ccc1Br C1(CC)CCN(C(=O)COCC2CC2)C1CNC(c1ccc(CO)o1)=O c1(CC)nc2sc(C)cn2c1C(N1CC(NC(=O)C(COC)COC)C(O)C1)=O C(=O)(C1=C(C)CCOC1)N1C(C(C(=O)NCCC=CC)(C)C)CCC1 C1(C(=O)Nc2nccc(C(=O)NC)c2)CC2CCC1N(C(c1ccn(C)n1)=O)C2 C1(NC(C(C2CCC2)OC)=O)CC(N=c2c([N+](=O)[O-])c[nH]c3c(Cl)cccc23)C1 C1(CCNC(=O)C(C2CCC2)C2CCC2)CN(C(C2CC2(F)F)=O)CCO1 C(=O)(C1SCCc2sccc21)C(c1[nH]c(=NCC)sc1)=O.C(CCOC)OCCN C(=O)(C1=CCC(F)(F)CC1)N1CC(CCCNC(Cc2cc(C)on2)=O)OCC1 c1(CC(N2C3C(NC(Cc4c(C)cccn4)=O)C(C3)C2)=O)nc(F)c(F)cc1F c1(C(=O)NC2(CN(C(c3cc(C)oc3C)=O)C)CC2)ccc(F)c(Br)c1 C1(CN(CCNC(=O)C(C)Cn2ccc(C)n2)CC)CCCOCC1 c1(C(N2CC(NC(C(CC)OC)=O)C(F)CC2)=O)cc(Br)c(C)cc1OC c1(C(C)NC(=O)NC2(CC)CCOC2)cnccc1-c1ccc(F)cc1 c1(NC(C(C2CCN(Cc3cccc(O)n3)CC2)C)=O)ccc(Br)cc1C(N)=O NS(=O)(=O)CCCC(=O)N1CC(O)(CNC(C23COCC2C3)=O)C1 CN=c1cc(C(=O)NC2CCCCC2CNC(=O)COCCF)cc[nH]1 c1(CC(N2CCC(N(CCC)C)CC2)=O)ccc2cc(OC)ccc2c1 C1(NC(C2C(C)C2)=O)CCN(C(=O)C(O)CC2CCCCC2)C12CC2 C(=O)(CC1C(=O)Nc2ccccc21)NC1CCN(C(C2(OC)CC2)=O)C1 C1(NC(=O)CNC(N2CCCC2)=O)CC2CN(CC3CCC(C4CC4)O3)CC12 c1(C(=O)NCCC2CCN(C(c3ccccc3)=O)C2)cc2cccnc2s1 Cc1cc(C(=O)NC2CC(NC(=O)CC3CCCOC3)C2)nnc1O c1(C(C(=O)N(CCN(C(=O)C(C)c2ccco2)C(C)C)C)C)ccc(F)cc1F Cc1cc(C(=O)N(C2CCCN(C(=O)CCCS(C)(=O)=O)CC2)C)cc(C)c1F CC(N=[N+]=[N-])C(=O)N1CCC(C(C)C(N2CCCC(C(N)=O)C2)=O)CC1 c1(CC)nn(C2CC2)cc1C(=O)N(C(C)CCNC(=O)CCc1cn(C)nn1)C C(=O)(C(C(C)NC(c1ccc(C)cc1)=O)C(C)C)NCCSCC=C c1(CNC(C(CC#C)O)=O)ccc(CNC(C23CCCC2(C(N)=O)C3)=O)c(F)c1 c1(C(=O)NC2(C)CN(C(C3(C)CCC(C)C3)=O)C2)cnc2c(c1)COC2 c1(C(N(C(C)C)CCNC(=O)C(F)(F)C(C)O)=O)noc2ncccc12 N1(C(c2c(N)ccc(C)c2)=O)CCOCC(C)(CNC(C2CC(N(C)C)C2)=O)C1 c1(SC)nc(-c2ccc(C(=O)NCCCO)cc2)sc1C C1(C(=O)NC(C2(O)CN(C(c3ccncc3F)=O)C2)C)CC2CC1CC2O c1(C(=O)NC2CCN(C(CC(C)n3ccnc3)=O)C2)cc(F)cc2nc(S)[nH]c12 C12(C(N(CCNC(C3C(C)(C)C3C#N)=O)CCOCCO)=O)CC3CC(CC(C3)O1)C2 C(CCCOC)(C(=O)NC1(CO)CCCCC1)NC(CCSCC(N)=O)=O c1(C(C)C)ccccc1CNC(=O)CC(O)CNC(=O)OC(C)(C)C N1(CC(=O)NCC2(NC(C3(C4CCC4)CC3)=O)CCOCC2)CCCCC1CO C(=O)(C(C(C)NC(=O)CCN(C)CCC)C(C)C)N(C)Cc1cccc(C#C)c1 c1(OC)ccc(F)c(C(=O)NCC2(C)CCCN(Cc3cccnc3)C2)c1 N1(C(CC2N(C)CC=CC2)=O)CC(NC(=O)Cc2ccn(C(F)F)n2)C(C)(C)C1 CCCCCCC(=O)N(CC)CC12CCC1CN(C(=O)CNC(=O)CC(F)(F)F)C2 c1(SCC(=O)NC2CCOCC2C(=O)Nc2cncc(O)c2)ccc(F)cc1 N1(C(C2CC(C)(CC)C2)=O)CCCCC1CNC(C1C(C(C)=O)C1(C)C)=O c1(OC)ccc(Br)cc1S(=O)(=O)N1CCC(N(C)C(=O)OC(C)(C)C)C1 C(=O)(C(C(C)NC(=O)CC1(NC(C)=O)CC1)C(C)C)NCCC(=O)NC C12(NC(C(C)CO)=O)CCCC1N(c1ccnc(-c3cccc(Cl)c3)n1)CC2 CN1CC(NC(=O)CC2C3CCC(C3)N2C(=O)OC(C)(C)C)CC12CCOCC2 c1(CCC(N2C(CNC(C(C)N(CC)CC)=O)CC2)=O)ccc(COC)cc1 c1(C(N2CCCN(COC(C3C(C)C3)=O)CC2)=O)cc(I)c(I)c(I)c1 c1(C(N2CCC(C)(NC(=O)CCc3cncnc3)C2)=O)c(O)cccc1F c1(OC)ccc(C(=O)NC2CC(CNC(c3cc(F)c[nH]3)=O)C2)cc1 n1(CO)cc(C(=O)NCCN)nn1.N1(C(C2C(C(=O)OC(C)=O)C2)=O)CCC1C c1(CCC)c(C(=O)NC(C)CN(C)C(c2cc(C)n(C(C)C)n2)=O)cnn1C c1(OCC)cccc(CNC(=O)CC2(c3ccon3)CCC2)n1 c1(N2CC(C)(NC(C(c3ccccc3)OCC)=O)C2)cc(Cl)nc(SCC)n1 c1(OCC(=O)NC2C(CNC(c3cccc(C)c3)=O)COC2)cc(F)cc(F)c1 C1(COC)(CNC(C2(F)CC=CCC2)=O)CCN(C(=O)C=CSC)C1 c1(CN(C(c2cnc(C)[nH]2)C(=O)NC(C)(C)C)C)cccn2nccc12 c1(CC)nc(C(C)Sc2ccco2)n(Cc2ccccn2)n1 C1(C)(C(=O)OC)CN(C(C)=O)CC1C.c12ccccc1-n1cc(nn1)CO2 Cc1ccc2c(C(=O)NC3(C)CCCN(C(C4CC(C)C4)=O)C3)onc2c1 CC1OCCN(C(C2CC(=O)CC(=O)C2)=O)C1C(=O)NCCc1ccns1 C1(C(=O)NCC2CN(C(C3(CCCC)CC3)=O)CC2(C)C)CCc2nncn2C1 N#Cc1cccc(OCC(=O)NC2CC3CC2N(C(=O)CN2CCCCC2)C3)c1 CC#CCCCC(=O)NC1CN(C(=O)CC)CC1(C)C c1(OC)ccc([N+](=O)[O-])cc1C(N1CCC(NC(=O)COCC2CC2)C(C)C1)=O c1(C(N(C(c2ccccc2Cl)C(=O)OC)C)=O)cc2n(n1)CCOC2 c1(NC(C2CCCN2Cc2cn(C(F)F)nn2)=O)cccc(COCCO)c1 C1(C(N2CC(CC)N(C(c3ccn(C)c3C)=O)CC2)=O)CCCC(F)(F)CC1 CC1(C)CC(O)(C(C2(c3cn(CC4C5CCCC45)nn3)CC2C)NN2CCCC2)C1 C#CC1(C(=O)NCCCCCN(C(=O)CCN(c2cnccn2)C)C)CCC1 c1(C(=O)NCC2OCCCN(CCC(C)F)C2)cc(F)c2ncccc2c1 N1(C(C2(CN(C)C)CC2)=O)CCCCCC(NC(C2CCc3nncn3C2)=O)C1 C(=O)(C1=CC2CCCCCC12)N(C(C)CNc1cnc(C#N)cn1)C CC1(C)CC(CS(=O)(=O)NCC(F)(C(=O)O)C(=O)O)OC(=O)N1 N1(C(C)C(=O)NCC2CCCC(=O)N2C)CCN(C2CCOCC2)C(C)C1 N1(C(C2CN(C)C(=O)C2)=O)CC(C)(C)C(NC(=O)CC(C)(F)F)C(C)(C)C1 CC1(C)OC(=O)CC1C(N1CC(C(=O)NCC(O)CF)C2(CC2)C1)=O c1(N(C=O)C(c2cn(C)nc2C(=O)C(F)(F)F)C)cc(C)cc(Cl)n1 C1(C(C)C)N(C(=O)CC2(N(C(=O)C=Cc3nccs3)C)CC2)CC1(C)C C1(CNC(C(CC#C)C)=O)CCC12CCN(C(c1nn(C)c(C)c1Cl)=O)CC2 C1(F)(CNC(c2c(-c3cn(C)nc3)cco2)=O)CCC(NC(C2CCCO2)=O)C1 C1(C)(C(=O)NC(C(C)NC(c2cc(OCC)ncc2)=O)CO)COC(C)(C)CO1 CC1(CNC(C2CC(=O)CN2C(c2c[nH]c(C#N)c2)=O)=O)CCCC1O CCCC(C)(CCC)C(=O)NC(CNC(c1ccnc(Cl)c1O)=O)C1CC1 N1(C(N(CP(C)(C)=O)CC(=O)O)=O)CCCC(C2CC2)CC1 C1(C(=O)NC(C)CN(C)Cc2ccc3nn[nH]c3c2)CCC2(CCCCC2)CC1 CN1CCN(C(c2cc(CC3CCC3)c[nH]2)=O)CC1CNC(c1cccnc1N)=O C=C1CCC(C(=O)NC2(C3CCCN3C(C3CCC(=O)C3)=O)CC2)CC1 Cc1ccc(NC(C2CC(N=[N+]=[N-])C2)=O)c(F)c1F c1(C(N(CCNC(c2conc2C)=O)CC)=O)nn2cccnc2c1Br C(=O)(C1=Cc2cc(F)ccc2OC1)N1C(C(C)NC(C2(C=C)CCC2)=O)CCC1 N1(C(c2csc(CO)n2)=O)CCOC2CCCN(C(C3(Cl)CC3)=O)C2C1 c1(NC(C)=O)ccccc1C(N1CC(Cn2cc(C3(F)CCOCC3)nn2)C1)=O O=C(CCCC1CCC1)NC1CCN(C(=O)CCC2CCCO2)C1 Cc1cc(F)ncc1C(=O)NC12CC(C(=O)Nc3cccc(C(C)(F)F)c3)(C1)C2 C(=O)(C(C)(C(F)(F)F)c1cc[nH]n1)NC1CCN(C(CCNS(C)(=O)=O)=O)C1 N1(C(c2c(CC)oc(C)c2)=O)CCC(O)C(NC(C2CN(S(C)(=O)=O)C2)=O)C1 C1(CNC(C2N(C(C)=O)CCC2)=O)CCCN(C(=O)Cc2ccns2)CC1 C(N=c1cc(C)nc(N2CCC(CNc3ccccc3)C2)[nH]1)c1cn(CC)nc1 N1(C(C(CC)OCC)=O)CCC2CCCC12C(=O)NCCCCOC(C)=O N1(C(c2cc(C)sc2-n2cccc2)=O)CC2CN(C(c3cscn3)=O)CC2C1 c1(OC)cc2c(cc1Br)CCN(C(=O)C(N1CCCC(O)C1C)=O)C2 Cc1cccc2c(C(=O)NC34CCN(C(c5ccc[nH]5)=O)CCC3C4)csc12 c1(N2CCN(CCCNC(C(C)(C)OC)=O)CC2)ncc2c(c1C#N)CCCC2 C(C(=O)NCC(F)F)(C(C)CC(C)C)N(CCOc1ccc(C)cc1)CC c1(C(=O)NCC2(F)CN(C(C3(C)CC3F)=O)C2)ccc2c(c1)CCCC2 C(=O)(C1=CC2CCC(C1)C2)NC1CN(C(C2(N(C)CCO)CC(O)C2)=O)C1 c1(C(=O)NC23CC(NC(C4C(C)(C)CC4)=O)(C2)C3)cc2c(cc1O)OCO2 CC(C)(CCC#N)C(=O)N1CC(NC(c2cnsn2)=O)C(O)C1 CCCC(CC(=O)N1CCC(OCCF)C1)NC(=O)CCC(C)(C)F C(=O)(CC1=CCN(C(=O)C2=CCCOCC2)CC1)Nc1cccc(N(C)C)c1 c1(C(C)=O)cccnc1NC.c1(C(N(CCCNC=O)C2CC2)=O)cnn(C)c1C1CC1 C1(NC(COCC=C)=O)CCCCN(C(=O)CN2CCC(C)(O)C2)C1 C1(C(N2CC(NC(=O)C=CC=C(Cl)Cl)C2)=O)(COCC)CCC1 C1(C(=O)NCC2CN(C(Cc3c(C)nccc3)=O)C(C)C2)COCCN1C=O c1(CC(C(=O)NCC(C)N(C(=O)CC2C=NN(C)C2=O)C)C)ccc(F)c(F)c1 C1(NC(=O)OC(C)(C)C)(CNC(N2CCOC(C3CCCOC3)C2)=O)CC(C#N)C1 N1(C(C(C(C)C)O)=O)CC2(CCC(CNC(=O)COC3CCCC3)O2)C1 C1(NC(c2c(OC)csc2)=O)C2CC3C1C3C2C(N1CCOCC(O)C1)=O c1(C(=O)Nc2c(COC)ccc(SC)c2)ccc2nonc2c1 N1(C(C(=O)NCCC2CC2)C2COC2)CCC(c2ccnc(O)c2)CC1 c1(C(=O)NC(CN(C(c2cc(COC)[nH]n2)=O)C)C)cccc2cnccc12 C(C)(C(=O)NC1CCCC1CNC(C1(C#N)CCC1)=O)(C1(C)CC1)OC c1(C(N2CCC(NC(c3ccc(COC)[nH]3)=O)C2C2CC2)=O)ccc(F)c(Br)c1 c1(C(N2CCCC(c3cn(CCCCCCO)nn3)C2)=O)ccc2[nH]ccc2c1F n1(C(=O)OC)cc(C(N2CCC2CC(C)C)=O)nn1.C12(CC1(C)C)C(=O)N2 CCCC(O)(CCC)CC(=O)NCCCC(C)NC(=O)C=Cc1ccc[nH]1 N1(c2[nH]c(N(C)C)nc(=NC)n2)CCc2ccc(OCCC#N)cc21 N1(C(c2c(CC)nn(C)c2Cl)=O)CCC2CCN(C(=O)C=CSC)CC12 CC(CCCCNC(C1CCC(=O)N1CCC(F)(F)F)=O)NC(=O)CCF Cc1cnc(C(=O)NCC(CO)NC(c2cc(C(C)C)oc2C)=O)nc1 C1(C(N(CC(=O)C(C)(C)C)C)=O)CC2(CCC1NC(=O)OC(C)(C)C)CC2 C(=O)(N=c1ccn(CC2CCCO2)[nH]1)Nc1c(C(N)=O)cc(-c2ccncc2)s1 C1(C(=O)OC)(CNC(C2CCN2C(C)=O)=O)CCOC1.C12C=CC(C1)C(=O)N2 C1(CC)CN(C(=O)C(C)(C)C)CCC1NC(=O)CCCSC C(=O)(C(CC(F)F)NC(C1CCCC(=O)N1)=O)NCCc1c(C)ncs1 C1(NC(=O)NC(C)Cn2cc(-c3ncoc3C3CC3)nn2)COc2ccccc2O1 c1(C(=O)NC(CN(C(c2ccccc2Br)=O)CC)C)cccc([N+](=O)[O-])c1 N1(C(C2CCC(C(=O)OC)C2)=O)CC2(CCN(C(c3cnc(O)s3)=O)CC2)C1 N1(C(CNS(NCC)(=O)=O)=O)CCOc2ccc(C(=O)OC)nc21 N1(C(C(C=C)C)=O)CCN(c2nc(CC3CC3)ns2)CC1.C(CCCC)N C(=O)(N1CCCc2nccn21)C1CN(C(C(C(C)(C)O)F)=O)CC(F)C1 c1(NCc2c(Br)cn(C)n2)[nH]c(=NCCCc2nc[nH]n2)nc2sccc12 C1(C(N(C(C)C)CCO)=O)CCCN1C(=O)C(C)C1CCCC1 c1(COCC)nc(-c2ccnc(N(C)C)n2)n(C2CCCc3ccccc32)n1 N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC(NC(c2csc(Cl)c2)=O)CC12CCC2 c1(C(N2CCC(NC(C(C)=C(C)C)=O)C(C)C2)=O)cccc2c1OCCN2C C1(C(N2CC(N3CCCC(C)C3)C2)=O)(OC)CCCN(C(=O)CC(F)F)C1 CC1Oc2ccccc2OC1CNC(=O)N(CC(F)F)Cc1ccccc1 N1(C(C(C=C)O)=O)CCC2(CCC2NC(=O)CCOCC(F)F)CC1 c1(OCC)ccc(CC(=O)NCC2CCN(C(=O)C(c3cnn(C)c3)O)C2)cc1 C1(CNC(C(CC2CCC2)OC)=O)CN(C(=O)C(C(C)C)NC(C)=O)CCC1(C)C Cc1nc(C(N2CC(C)(C)C2c2ccccc2)=O)c(C)n1C CC1CCC(CC(N2CCC(N(c3nccc(CC#N)n3)C)C2)=O)CC1 C1(C(=O)N(C2CCCN(C(C3CCCCC3)=O)C2)C)CCC2(CC1)CC2(F)F c1(C(C(=O)NCCOC)N(C)CC2(C#N)CCC2)cc(Cl)c(F)c(Cl)c1 CN1N=C(C(=O)NC2CS(=O)(=O)CC2NC(=O)C2=CCCC2(C)C)CCC1=O C=CCC(C)(C)C(=O)NCC1CC(NC(=O)C=CCN2CCOCC2)C12CCC2 c1(C(N2C(C)(C)CC(CNC(C3(F)CCCOC3)=O)C2)=O)cccc2nncn12 C1(NC(c2cc3scnc3[nH]2)=O)CN(C(=O)COCC2CCOC2)CCC1F C(CNC(C1CCC1)=O)(CO)NC(=O)CSc1nccs1 C1(C)(NC(C(CCN(C)C)OCCNC(C)=O)=O)CC2(C1)CC2(F)F.C1C(=O)O1 N1(CC)C(=O)CCC1C(=O)N(C(C)CN(C)C(c1cc(CF)on1)=O)C CC1(C)CCCC(NC(C23CC(CO2)N(C(c2cnnn2C2CC2)=O)C3)=O)C1 N1(C(c2cnc(C(C)=O)s2)=O)CCC(NC(c2csc3nnsc23)=O)C1(C)C c1(C(=O)NCc2c(C(N(CC(=C)C)CC)=O)[nH]cc2)cc(F)n(C)n1 c1(-c2ccn(C)c2)ccc(CNCc2cccnc2N2CCCCC2)cn1 c1cc2cc(CN3CCC4(CCO4)C3)ccc2nc1N1CCN2CCCCC12 O(N(CC)C(=O)CN(C(C)=O)CC)C(C1CC(=O)C1)=O c1(NCC(CCCC)NC(c2oc(CC)nc2C)=O)ncc([N+](=O)[O-])cc1Cl N1(C(C=CC(=O)OCC)=O)CC(NC(=O)C(C)(C)CO)CC1CO C1(c2n(CCOC)nnn2)(NCC2CCC(C)C2)CCN(C(C)=O)CC1 C1(C(N2CCCC2C(=O)O)C(=O)NCC)COC(C)C1.c1(C)ccsc1 O=C(C1CCc2ccccc21)NCC(C1CCCC1)NC(C1CC(=C2CC2)C1)=O N1(C(C(c2ccc(C)o2)C)=O)CCC(C)(C)CC1C(=O)NCC(C)(C)CN=[N+]=[N-] C(=O)(CC(C)(CC)C(=O)OC)N1CCN(CCNC(C(CCC)=CCC)=O)CC1 C1(C(N2C(C(N3C(CC)COCC3)=O)CCC2)=O)CC2C=CC1CC2 Cc1ncncc1C(N1CC(OCCC(N2CCC(C(C)O)C2)=O)C1)=O C12(CNC(=O)NCC(C3CCOCC3)O)CC(NC(=O)C3CC3)(C1)C2 C1(CNC(CC2C(C)OCC2)=O)CCC(N(C)C(c2cc(CO)ccn2)=O)CC1 c1(C(=O)NCC(CNC(c2nnc(CC)s2)=O)O)ccc(F)c2ccoc12 C=C(I)CC(=O)NCC(O)CCNC(=O)CCC1CCCC1 C12(CNC(c3cc(-c4ccco4)c[nH]3)=O)CN(C(C3C=CCC3)=O)CC1CCO2 c1(C(=O)NC2C(NC(C(C)NS(C)(=O)=O)=O)CCOC2)sccc1S(N)(=O)=O C1(OC)CN(Cc2ccc(O)cc2)CCC1NCc1ccccc1NC(C)=O C1(C(=O)NCC(CO)NC(c2cccc(S(C)=O)c2)=O)CCC2(CC1)CC2(F)F c1(NC(C2CC(O)CN2Cc2cccc(Cl)c2)=O)nc(O)nc(O)n1 S(=O)(=O)(c1cc(Br)cc2cccnc12)OCOC(C1CCCCC1)C Cc1cnc(C(=O)NCC2CC3CN(C(C4(n5ccnn5)CC4)=O)CC23)cc1C C(=O)(C1=CCCCC1C)NC(CSCC)C(=O)NCCN1CCCC1C N1(C(=O)NCC2(CC)CCOCC2)CCC2(CC(C#N)C2)C1 Cc1cc(CN2C3CC2CN(C(=O)C=Cc2ccc(Cl)cc2)C3)c(C)cc1Br c1(C(N(C(C)C(=O)N(C)CC2(CO)CCC2)CCC)=O)sc(C)cc1C N1(c2cc(NC3N(C)CC3)ncn2)CCc2c(-c3ccc([N+](=O)[O-])s3)cccc2C1 C1(C2CC2)(C(=O)NC(CC)CNC(c2nc(C3CC3)ncc2Cl)=O)CCOCC1 Cn1ncc(Cl)c1CC(=O)NCC1CC1NC(=O)Cc1cc(Cl)n(C)n1 C(C(CO)NC(C1(C)CC1)=O)N(C(=O)COC1CC1)OCC.C(CC(C)C)OC c1(CCC(=O)NC(CC)CNC(c2cnc(C3CC3)[nH]2)=O)c(C)nc(O)nc1C c1(SCC2(C(=O)NC3CCC3NC(=O)C(F)(F)C3CC3)CC2)ccccc1Cl C1(CC#C)(C(=O)NCCC(C)CO)CCN(C(=O)CC(C)CC)C1 C(C(CNC(=O)Cc1cncn1C1CC1)CO)NC(C1CN(S(CC)(=O)=O)C1)=O N1(C(C(C)(C(C)C)NC(C)=O)=O)CC2CCN(C(=O)C=C(Cl)Cl)C2C1 N1(C(C2(C#C)CCC2)=O)C2CCC(C2)C1C(=O)NCC(C)OC C1(SC)CCN(C(=O)CCCNC(=O)C(O)C2CCCC2)CC1 N1(C(CCSC)=O)C2CCC1CN(C(C1CC1c1cc(F)ccc1Br)=O)C2 Cc1ccc(Br)cc1CC(=O)NC1CCC1c1ccccc1 c1(OC)cccc(CC(C)CC(=O)NC(C)CN(C(=O)CCc2nc[nH]n2)C)c1 C1(C(=O)NCC2CN(C(C3N(C(C)C)C(=O)CC3)=O)C2)CCOC2(CCC2)C1 C(C(=O)NCCCN(C(=O)CC1CCC(O)C1)C(C)C)(C(C)C)OC c1(CCNC(C(CNC(c2cc(C(N)=O)[nH]n2)=O)O)=O)cccc(F)n1 C(N=c1[nH]c(NCC2CC(=C3CCC3)C2)nc2ccsc12)c1nnc(C)o1 C(=O)(C1=CCC(C)CC1)N(CC(CNC(C1(OCC)CCCC1)=O)C)C C(=O)(C(C(=O)N1CCCC(CCNC(=O)CSCC(C)C)C1)C(C)C)OC C1(O)(C(C(=O)NC(CN(C(c2nn(C)cc2C)=O)CC)C)(F)F)CCCN(C)C1 c1(C(=O)NC(CC(C)NC(CC)=O)C)cc2c(OC)cc(F)cc2[nH]1 C(CCCCCNC(C1C2CC2C2CC12)=O)NC(=O)C=Cc1ccsc1 c1(C(=O)NCC2N(C(c3ncn(CC)n3)=O)CCC2)cc2cccc(OC)c2o1 Cc1cc2sc(C)c(NC(N3CCC4CN(C(=O)OC(C)(C)C)CC34)=O)c2cc1C c1(C(=O)OCC)sc2ncc(Br)cc2c1NC(C1CC2C=CC1O2)=O C1(c2nnnn2C(C)(C)C)(NCC(c2ccccc2)C)COC2(CCC2)C1 C1(CC(=O)NCC2CC2CO)CCCN(C(=O)CC23CCC(CC2)C3)C1 Cc1noc2ncc(C(=O)NC(CNC(c3ccc(S(C)(=O)=O)s3)=O)CO)cc12 CC1=C(C(=O)NC(C)(C)CCNC(=O)C(F)(F)CO)CCO1 C(C)(CC(C)(C)C)NC(CC1N(C(C2C(=C)C2C(=O)OC)=O)CC1)=O c1(C(=O)NC2C(NC(CC3CC(OC)C3)=O)C2)cnc(O)n(C2CC2)c1=O C(CC(C(C)(C)C)NC(=O)CSC(F)F)N(C)C(C1CCC(=O)NC1)=O N1(C(CC(CC)SC)=O)CCCN(C(C2(Oc3cccc(C#N)c3)CC2)=O)CC1 c1(C(=O)NCC2CC2NC(C2CCCCC2)=O)cncc2c(Cl)cccc12 Cc1ccc(Cl)cc1C(N1CC(NC(=O)C(C)Cn2cccn2)C(C#N)C1)=O c1(C(=O)NC(C2CN(C(=O)C3=CC(C)(C)C3)C2)C)ccc2nncn2c1 c1(C(N2C(CC)CCCC2C)=O)cc(-c2cccc3c2OCC3)c2n[nH]cc2c1 c1(C(N2CC3(N(C(CCNC(N)=O)=O)CC3)C2)=O)ccc2cnoc2c1 C1(C(N2C(CNC(CC3CC(C)C3)=O)CC(C)(C)C2)=O)COc2ccccc2O1 c1(OC)ccc(C)c(C(=O)NC(CNC(=O)CC2CC(C)=NO2)C2CC2)c1N c1(OCC(N2CC(N3C(=O)CC(NC4CC(C)C4)C3)C2)=O)cccc(Cl)c1Cl CC(CC(=O)NC1(C)CC(NC(=O)C(C)(C)C2CCCCC2)C1)C1CCCC1 c1(OC)ccc(-c2cc(C(N3CCCC3C(=O)Nc3ccccc3)=O)n[nH]2)cc1 C1(CNC(=O)C=CCN2CCC2)(CO)CC12CCN(C(C1CCC3(CC3)C1)=O)CC2 c1(C(=O)NNC(=O)c2ccc(N3CCCNC3=O)cc2)ncc(Cl)cc1Br N(C1CS(=O)(=O)Cc2ccccc21)C(C(C)NCCC)=O.c1ccccc1 c1(NC(=O)Nc2cnn(C(C)C)c2C2CC2)nccc(I)c1F C1(COC)CN(C(c2cc(C(N)=O)cn2C)=O)CCN1C(=O)COc1ccsn1 C(=O)(C(CC)C(C)C)NCC1(C(=O)NC(C(=O)OCC)CC)CCCC1 C1(N(C(C(=O)NCC)=O)C)CCC(NC(c2csc(CSC)n2)=O)CC1 c1(NC(C2(CCOC)CCNC2=O)=O)cc(Br)cc2c1OCO2 N1(C(c2cn(C)nc2)=O)CCC2CN(C(=O)CCS(C)(=O)=O)C2C1 CCC(C(=O)N(CC(C)NC(=O)CSCC(C)C)CC)n1ccnc1 CC1CCN(C(CC2(C)CCOC2)C(=O)NCCN2CCOCC2)CCS1 c1(C(N2C(C(=O)NCc3cc(C)nc(C)c3)C=CC2)=O)cccc2cc[nH]c12 CN1CCC(CC(=O)NCC2(NC(=O)CC3CCN(C)C3=O)CCOC2)CC1 N1(C(=O)COC(F)F)CCC2C(C1)CN2C(=O)Cc1ccc(Cl)c(Cl)c1 C1(NC(C(C)O)=O)CCN(C(=O)C(Cc2ccccc2)n2cnnn2)CC1(C)C C1(CC(=O)NC(C)(CNC(c2cnn(CCO)c2)=O)CO)SC2=NCCN2C1=O Cc1cc2[nH]c(C(=O)NCCC3(NC(=O)CCc4cnc(O)[nH]4)CC3)cc2s1 c1(C(N(C2CC(NC(C(CCOC)(C)C)=O)C2)C)=O)ccc(F)c(F)c1N FC(F)(F)C(CN=c1[nH]c(N2CCC(n3cccn3)C2)nc2ccsc12)C1CC1 c1(CC(N2C(CNC(c3ncccn3)=O)C=CC2)=O)ccc(Cl)c(F)c1 C(=O)(CCCC(C)=O)NC(C(C(C)C)NC(c1cnc(CC)nc1)=O)C c1(C(N2C(C)(C(=O)Nc3cccc(Cl)c3I)CCC2)=O)n[nH]c2c(Cl)cccc12 C1(C)(C(N(CC(O)CNC(=O)CN(C)C2CC2)C)=O)CC2CC2C1 C12(C(N3CCC(c4nn[nH]n4)C3)=O)CCCC1N(C(c1cnc(Cl)s1)=O)CC2 C1(C(=O)NCCN(C)CCN(C)C)CCCCC1NC(C1(C)C=CCC1)=O CCC(CC)CC(=O)N1C(CC(=O)NCC(C)CN(C)C)C2CCCC12 C1(C(N2CC(CC(=O)N(CC)Cc3cccnc3)C2)=O)CCC(C2CC2)C1 c1(C(=O)NC(C2(C(=O)NCC3(CO)CCOC3)CC2)C)ncccc1O C1(CC(=O)NCCCC(C)NC(c2[nH]cc(C)c2)=O)CCCC2(CCC2)O1 C1(CNC(C2CC2C(F)(F)F)=O)CCN(C(C2(C(F)(F)F)CCCCO2)=O)CC1 O=C(C1=CCCC1)NC(Cc1ccco1)C(=O)NCCC(=O)N1CCCC1 c1(C(N2C(COC)CN(C(C3CCCN3C)=O)CC2)=O)cc(C)cc([N+](=O)[O-])c1 c1(C(N(CC(O)CNC(=O)CNC(N)=O)C)=O)ccc(-c2ccco2)[nH]1 C(=O)(C(O)CC(C)(C)C)NC(c1cccc(C)c1)CNC(=O)Cn1ccc(C)n1 c1(CC)cc(C(=O)N(CCCNC(=O)C(C)(C2CCOCC2)OC)CC2CC2)n[nH]1 N1(C(C(CC)c2ccccc2)=O)CCC(NC(c2cc(C(C)(F)F)on2)=O)C1C C1(CNC(C2C(C)C2)=O)CC12CCN(C(=O)COC1CCCC1)CC2 CC(C(=O)NNc1ccc(-n2ccnc2)cc1)c1ccc(S(C)=O)cc1 C1(C(=O)NCCC(CC)C)CCC(CNC(=O)CCCn2ccnn2)CC1 N1(C(CCc2n(C)cnc2)=O)CC(NC(C2CCC(NC(N)=O)CC2)=O)C2(CC2)C1 c1(CN2CCC(O)(C(=O)NCc3ccc(C(C)C)cc3)C2)cc(F)cc(Br)c1F C(=O)(C(=O)N=S(C)(C)=O)N1C2CCC(NC(C(C)C#N)=O)(C2)C1 S(=O)(=O)(c1cccnc1)N(CC(N1C(CNC(CCC=CC)=O)CC1)=O)C C1(CNC(Cn2nnc(C)n2)=O)COCCN(C(C2CN(C(N)=O)CCO2)=O)C1 C12(NC(C3N(C)CCC3)=O)CC1CN(C(=O)Cn1ncn(C)c1=O)C2 CCC(CN(C)C)C(=O)N1CCC(CCNC(=O)Cc2cnn(C)c2)CC1 C1(CNC(C2C(C)C(=O)C2)=O)CC2CCC(C1)N2C(c1cccnn1)=O C(=O)(C(C)(O)C(F)(F)F)N1C(C(N(OC)CCCO)=O)CC2(CC2)C1 NS(=O)(=O)CC(=O)NC1CC(NC(c2ccc(CCNC(C)=O)o2)=O)C1 c1(CNC(c2cc(SC)no2)=O)cccc(C(=O)NC23CC(C(N)=O)(C2)C3)c1 c1(CN(CCNC(CC)C(N)=O)CC)ccc(F)cc1Br CCC(C)(CNC(C1CC1(C)C(F)F)=O)C(=O)NCc1nn(C)cc1CO C1(NC(c2c(C)nc(C)s2)=O)CCC2(CC1)CC(NC(C1CC1C)=O)C2 Cc1cccnc1CC(=O)NCc1ccc(CNC(=O)C(C(C)O)N(C)C)cc1 C1(C(=O)NCC(COC)(F)F)CCC2CCC1N2C(=O)Cc1cnn(C)c1 C(C(=O)NC1CCC(CNC(c2sc(SC)cc2C)=O)CC1)(C(C)C)SC c1(C(=O)NC(CCNC(Cc2c(OC(C)C)cccc2)=O)C)c(N)cccc1F c1ccc(-n2cncn2)c(-c2ocnc2C(C2(CO)CC2)NC2COC2)c1 c1(NCC)c(F)cc(I)cc1F.Cc1cnc(C(=O)OC)c(F)c1.c12cccnc1CN2 C(CC(C)C)(C(=O)NCC1CN(C(C2CCCC(C)C2)=O)CC1(C)C)OC Cc1cc(NC2CCCN(C)C2)ncc1S(=O)(=O)NC(C(C)C)C(C)C C1(NC(C2(CCOC)CC2)=O)CN(C(c2cccc(C)c2C)=O)CC2CC12 Cc1nc2cncc(C(=O)NCC3(C)CC(F)(F)CN3C(c3ccoc3)=O)c2[nH]1 c1(OCC(=O)NCCC(C)N(C)C(c2cccs2)=O)cccc(F)c1 c1(C(N2CC3C(NC(c4c(C)sc(O)n4)=O)(CC3)C2)=O)ccc2c(c1)CCCO2 Cc1cc(CNC(=O)CC2CCCC2C)oc1C(N1CCC(O)(C(F)F)C1)=O N1(C(N(CC(C)OC)C)=O)CCC(CNC(C2(C(=O)N(C)C)CC2)=O)CC1 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC1CCC(NC(C2C(CC)C2)=O)C1 c1(OC2CCN(c3ccc(CCN)cn3)C2)c(Cl)cc(Cl)cc1Cl N1(C(CC=C)=O)CCN(C(c2ccn(CCF)n2)=O)C(CC(=O)NC)C1 c1(-c2cc(OC)c(C)cc2)nc(C2CCc3nnc(C)n32)n(CC(C)CO)n1 C(=O)(C1=CCCCC1C)NCC1CC(NC(C(C(=O)OCC)C2CC2)=O)C1 CCC(N=c1ccnc(NCCc2nc(=N)s[nH]2)[nH]1)c1cc(C)ccc1C C1(NC(=O)Nc2cnn(CCO)c2)CC2CC(C1)N(Cc1ccc(Cl)cc1)C2 Cc1nc(CCC(=O)N(C2CN(C(=O)C(C)(C)C#N)CC2F)C)[nH]c1C C(=O)(C(COC)CC(C)C)NCC(C(C)C)NC(c1c(NC)snc1C)=O C1(C(N2CC(C#C)(C(=O)NCC(C)SC)C2)=O)CC(=O)N(OC)C1 c1(CN(c2n(CCC=C)c(Cc3c(C)noc3O)nn2)C)c(F)cccc1Cl c1(C(N(C2CCN(C(c3n(CC#N)ncc3)=O)C2)CCO)=O)cc2ccsc2s1 c1(C(N2CC(C)(NC(c3ccc(F)c(F)c3N)=O)C2)=O)ccnc2c1ccn2C c1(OC)cc(CS(C)(=O)=O)ccc1C(=O)NCc1ccc(OCCO)nc1 C1(NC(C2CC(C#C)(O)C2)=O)CCC2CCN(C(C3CCC(F)C3)=O)C1C2 C1(C)(CC)CCCC1C(=O)OCC.N1(CC(=O)NCCNC)CSCC1=O CS(=O)(=O)c1ccc(C(=O)NCC2COCCN2C(c2cc(C(N)=O)co2)=O)s1 N1(C(C2CC(C(C)=O)C2(C)C)=O)CCC(C)(C)C1CNC(=O)Cn1cccn1 C12(C(N(C3CCCN(c4nccc(C(C)(C)C)n4)C3)C)=O)CCCCC1C2(F)F c1(CC)nc(C)c(C(=O)NC(C)(CNC(C2CCC(N(C)C)CC2)=O)CO)s1 C1(C(=O)NCc2ccc(SC)cc2)CCN(C(c2ccc(F)c(O)c2)=O)C12CC2 CC1CN(C(=O)CN2C(=O)CN(C)C2=O)CCC1N=c1cc(C(N)=O)nc(Cl)[nH]1 CC(C)CC(C(=O)NC1CCN(CCCO)C1)N(C(=O)CC1NC(=O)NC1=O)C N1(C(C2C(=C)C2)=O)C(CNC(=O)Cn2ccc(CC)n2)CC2COCC12 N1(C(CCCO)=O)CC(C)CCC1CNC(=O)CN(C)CCO.C(COCCO)OC C(CC(=O)N1CCN(CCNC(c2cc(C#N)n(C)n2)=O)CC1)(C(C)C)OCC C12(C(N(C(C)C(=O)NCc3ccncc3)CC3CCCC3)=O)CCC(CC1=O)C2 Cc1cc(C(C)NCc2ccc(N3CCCS3(=O)=O)c(F)c2)c(O)cc1Cl N1(C(C2(SC)CC2)=O)CCCC2(CCN(C(=O)CC3CC(SC)C3)C2)C1 C1(C#N)(CCN(C(CCC2(C#N)CC2)C(=O)Nc2ccccc2)C)CCOCC1 N1(C(C(C=C)(C)C)=O)CCN(C(c2nc(CC)oc2C)=O)C(C2CC2)C1 C1(CNC(C2CC(CCN3CCC(c4cnn[nH]4)C3)C2)=O)CCCC1C(CC)=O CC(C)(CNC(C1CC(F)(C(=O)OC)C1)=O)CC1CN(C(=O)CSCCF)C1 c1(C(N2CC3(CC(NC(c4c(O)cc(C)nn4)=O)C3)C2)=O)scc2c1OCCO2 CC(C)C(O)C(F)(F)C(=O)N1CCN(C(c2cn(C3COC3)nn2)=O)C(CF)C1 N1(C(C(=O)Nc2ccc(C)s2)=O)CC2(CC(NC(C3CCC4(CCC4)C3)=O)CO2)C1 c1(C(=O)NC(C)C(C)(C)NC(=O)CC(C)n2cccn2)ccc(O)c(CO)c1 c1(OC)ccc(C(=O)NC2CC(C)CN(C(c3nnn(C)c3C)=O)C2)c(F)c1 C(=O)(C1=CCN(C(C)=O)CC1)NCC=CCNC(CN(C)C(C1CCCC1)=O)=O C1(O)(CCNC(=O)NC2(CN)CCC2)CCOC1 N1(C(C(C)OC)=O)CCC(CCCCCNC(c2cccc(C)c2)=O)CC1 C(=O)(C(C)S(C)(=O)=O)NC(C(=O)NCc1c(OC)cccn1)(C)C1CCC1 C1(CCC=C)(C(N2CCC(CNC(C3CSCCS3)=O)C2)=O)CCCC1 C#CCCC(O)C(=O)NC1CCC(NC(=O)CCC(CC)OC)CC1.C(C)(C)(C)OC=O C1(NC(CC(CC)(O)c2ccccc2)=O)CCc2nc(NC(=O)CSC)sc2C1 Cc1[nH]nc(Cl)c1C(N1CCC(N(C)C(c2nnn(C(C)(C)C)n2)=O)C1)=O N1CCC2C(C(N)=O)C2C1.C1C(O)CC(=O)NC2(CC(=O)NO1)CCC2.CNC C(CN=c1[nH]c(=NCC2CC2)c2cc(C(F)(F)F)ccc2[nH]1)C1CC(C)OCC1 Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCCC(NC(C2(C)CC=CCO2)=O)C1 N1(C(C(C)(C)SC)=O)CC=C(CNC(C2Cc3cscc3C2)=O)CC1 c1(N2CCC(OCCOCC)C2)nc2ccsc2c(=NCCC(C)OC)[nH]1 C#Cc1cc(C(N2CCC(N(CCO)C(c3ccc(N)cn3)=O)C2)=O)cc(F)c1 N1(C(C2CCN(C)C2=O)=O)CCC(NC(=O)CCCCF)C2(CCC2)C1 CCCC(C(=O)N1CCSCC1C(N1CCC(CC(=O)OC)C1)=O)OC CC1CCN(C(=O)C(c2ccccc2)F)CC1CC(N1CCCC1CC(N)=O)=O C=CCC(C)(CC)C(=O)NCCN(C(=O)CCCOc1ccccc1C)C C#CC1(C(=O)NCCC2CC(C)(C)CO2)CCN(C(c2cc(CC)n(C)n2)=O)C1 c1(N2CC(CCNC(C=C)=O)C(F)C2)nc(S(C)(=O)=O)ncc1F Cc1cc(Cl)c(Cl)cc1C(=O)NC1CC(CNC(c2cnc(=N)[nH]c2)=O)C1 c1(OC)ccc(CCC(=O)NCC23CC2CCCN3C(C)=O)cc1Br c1(C(=O)NC(C2CCCCN2C(=O)C(C)CC(N)=O)C)nc2cccnc2s1 CC1CC(C)N(C(C2CC3C=CC2C3)=O)CCN1C(C12CCC(CC1)C2(C)C)=O c1(C(N2CCCC2c2cn(Cc3cccnc3)nn2)=O)ccccc1I c1(SCC(=O)N(C)CCNC(C23CC2COC3(C)C)=O)nccc2ccccc12 Cn1cc(C2=NOC(C(=O)NC(C)CCNC(=O)Cn3ncc(Br)n3)C2)cn1 C(=O)(CC(O)CNC(=O)CCc1nc(O)n[nH]1)NC1(C)CCOC1 N1(C(CC(=O)NCC2CC2)=O)CC2OCCN(C(=O)C(O)CC(F)(F)F)C2C1 N1(C(COCC#C)=O)CCCC(NC(C2CCC2(F)F)=O)C1CC c1(C(N2CC(C(C)NC(C3C4CCCC34)=O)C2)=O)cc2n(n1)CC1(CC1)C2 C1(O)(CCn2cc(-c3c(C)ncs3)nn2)CCN(C(C2(C(F)(F)F)CC2)=O)CC1 C1(C(=O)NC(c2onc(CC)n2)C)C2CC3C(C2NC(c2ccon2)=O)C13 CCCC(C)(O)C(=O)NCC1CCCCC1NC(=O)C1=CCCCC1 CC1CN(C(C2(C)CCCN(CC3(C#N)CCOCC3)C2)=O)CCN1C C(=O)(C1c2ccccc2CN1C(=O)OCC)OC Cc1cc(N2CCC(NC(N3CCC(CO)C(C)C3)=O)CC2=O)nc(C2CC2)n1 C1(CC(=O)NCc2c(CC)cccc2)CC2(C1)CN(C(C1CC1(C)C)=O)C2 C(=O)(C1CCCc2ccccc21)OCC1C(C)CCC1 c1(CN(C(C=CC(C)NC(C(=O)NCC)=O)=O)C)ccc(C)cc1 Cc1nc(C)n(CCCC(N2CCC(O)(C(F)(F)F)C2)=O)n1 C1(CC(=O)NC)CN(C(=O)COC2CCCC2)CCN1C(c1cc(SC)no1)=O CC1(NC(=O)CCC2NC(=O)NC2=O)CCN(CCn2ccc(C3CC3)n2)C1 N1(S(CCCC)(=O)=O)CCC2(CCN(C(C3CCC(C(=O)OC)CC3)=O)C2)C1 N1(C(c2cn(CCO)nn2)=O)CCCN(C(c2cc(CO)ccn2)=O)C(CO)C1 c1(C(=O)NCCN(C(C2(CC#C)CC=CCC2)=O)C2CC2)ccc(F)c(OC)c1 c1(C(=O)NCCN(C(CCN(C)CC)=O)CC)ccn(CC(F)(F)F)n1 c1(CN(C(c2ccc(F)cn2)C(=O)NC2CCOCC2)CC)ccc(F)cc1F c1(N2CCC(CNC(C(C(C)(C)C)=O)=O)C2)ncnc2cc(Br)ccc12 CC(O)CCCNC(C1CC1CNC(=O)CC1CC1)=O c1(C(N2CCC(NC(c3c(C)onc3)=O)C(C)C2)=O)cc2ccccc2o1 c1(CC(=O)NCCCC(C)NC(c2cc(F)ccc2F)=O)ccnc(F)c1F C1(C(=O)NCC2CCN(C(c3cncc(Br)c3)=O)C2)CC2CCC(C1)O2 N1(C(c2c(C)ccc(O)c2)=O)CCC2(CC1)CN(C(=O)C(C)OCC(F)(F)F)C2 N1(C(CCNC(C)=O)=O)Cc2nccnc2CC1C(=O)Nc1c(Cl)ccnc1Br N1(C(=O)NCC2C(CC)C2)CCCCCC1c1ccc(C)o1 c1(N(C)CCO)ccc(CC(c2csc(=N)[nH]2)=O)cc1.c12ccc(s1)CNCC2 CCC(C)C(CO)NC(C1CN(C(C2CCC(C(=O)OC)CC2)=O)CCN1)=O c1(C(=O)NC(C(C)C)CCN(C)C(C2CCCN2C)=O)cnc2ccnn2c1 C1(NS(CCOCC#C)(=O)=O)CC(C2CC2)(OC)C1 c1(C(=O)NCCC2(O)CCN(C(=O)CC3(O)CCC3)C2)cnc2occc2c1 C#Cc1ccc(C(=O)NCCSCC(=O)NCC2CCCCC2F)nc1 CCC(CC(=O)N(C1CN(C(=O)C(C(C)C)n2cnnn2)C1)CC)C(C)(C)C N1(C(C2(C)CCC(=O)N2)=O)CCCN(C(=O)CC2(O)CCCCCC2)C(CO)C1 c1(C(=O)NC(C2CCN(C(C3C(=C)CC3)=O)CC2)(C)C)nccc2ccncc12 c1(C(N2CC(NC(=O)CCc3ccc[nH]3)C2)=O)coc(CC2CC2)n1 CCC(C)CCCCC(=O)N(C(C)CNC(c1cccc(Br)c1N)=O)C N1(C(c2nc(C)[nH]n2)=O)CCC(C2CCCN(C(C3CCCOCC3)=O)C2)CC1 N1(C(CC(C)(C)O)=O)CCCC12CCCN(C(=O)C(F)C1CCOC1)C2 N1(C(c2ccn(CC)n2)=O)CCC(COC)(NC(C2(C)COCCO2)=O)CC1 C1(C#N)(C(=O)NC(C(C)NC(c2ccc(CO)cc2)=O)C)CCCOC1 N1(C(CC2C(C)C2)=O)CC2(CCN(C(=O)Cn3cnc(C(N)=O)n3)CC2)C1 c1(C2C(C(N(CCNC(=O)C(C3CCCO3)C3CC3)CC)=O)C2)ccncc1F C1(C2(NC(C3(C(C)NC(=O)CC=CC4CC4)CC3)=O)CC2)CCCO1 N1(C(C2(CC#C)CC=CCC2)=O)CC(C2CCN(C(=O)C(C)C(C)O)CC2)C1 C(=O)(NNc1ccnc(O)c1)NC(CC)(C)CCC(=O)O C1(C(=O)NC(C2N(C(C=COCC)=O)CCC2)C)CC2(CCOC2)C1 CC1C(C(=O)N(C)CC(C)(C(=O)N2CCC2(C)C2CC2)C2CC2)CCN1C C1(N(C)C(=O)N)CCCC(CCC(F)(F)F)C1.c1(COC2COC2)ccnc(N)c1 CC1=NN(C)C(=O)C1C(N1CCC1CNC(c1ccc(C2=CC=COC2)s1)=O)=O C1(NC(c2ccc(CC)c(Cl)c2)=O)CC2CCC(C1)N2C(c1cccs1)=O C(=O)(CP(=O)(C(C)C)C(C)C)NC1CCN(C(CSCC)=O)CCC1CO CCCC(C)CC(=O)N1CCCC1C(C)(C)CNC(C1CC(=O)N1)=O c1(C(=O)NCCCCC(=O)N(c2c[nH]ccc2=O)C)cccn2cncc12 C(=O)(CC(C)(C)CN(C)C)N1CC(CC(=O)NCCC(C)N(C)C)OCC1 N1(C(CN(C)C(=O)C2CC2)=O)CC2OCC(NC(=O)CCC3CC(C)(C)CO3)C2C1 C=CCC(CNC(=O)C=C(C)COCC)C(=O)NCCOCCO C1(F)(C(C)(C)O)CCN(N2CC(O)(C(CNC(C3CCC4CC34)=O)(C)C)C2)C1 C1(C(=O)NC2CCN(C(c3cc(-c4ccns4)on3)=O)C2)CC2C=CC1C2 C1(C(=O)NC(CN2CCN(C(C3N(CC)CCC3)=O)CC2)C)C(F)(F)C12CCC2 c1(C(N2C(CCNC(CS(=O)(=O)N(C)C)=O)CCCC2)=O)cccc2c1OCO2 C(CN=[N+]=[N-])(C(=O)NC(c1ccncc1)C)NC(c1cnc(C)o1)=O C1(C(=O)NCCn2cc(C(=O)NCC(C)CC3CCC3)nc2)CNC(=O)CC1C C(C(=O)N1CCCc2nccn21)C1CCN(C(C(C(C)C)S)=O)CC12CC2 C1(CC#C)(C(=O)NCC(CC)NC(=O)Cc2cscc2Br)CCCO1 c1(N(C(C(C)O)=O)CCNC(=O)COC2CCCC2)cccc(Cl)c1 N1(CCC)C(=O)CCC1C(=O)Nc1ccc(-n2cccc2)cc1 c1(C(C)NC(=O)Nc2nc(C(=O)OC)c(Br)[nH]2)cnc(O)c(C(F)(F)F)c1 C(=O)(CC1COc2cc(O)ccc21)c1c(F)c2ccc(C)cc2cc1 C1(C#CC(=O)N(C2CCC(CNC(=O)CC(C)n3cccn3)CC2)C)(CC)CC1 CCCC(CCCNC(=O)C(C)(O)CC(C)C)NC(c1coc(Br)n1)=O C1(CNC(C2CC(C)N(C)C2)=O)CCCCCN1C(c1coc(C(F)(F)F)c1)=O C1(NC(C(CSC)C)=O)CC(F)CN(C(=O)COCC2CCC2)C1 C(=O)(C(C)(O)C(C)C)NC1CC(F)(CNC(C2N(C(C)=O)CCC2)=O)C1 c1(-n2cc(C)nn2)ncc(Cl)cn1.CCC(C(=O)OC)N(N(CC(COC)C)C)CC C1(CNC(C=C(CC)C)=O)CCCCCN1C(=O)CC1CCCSC1 c1(C(N2C(CC)CCC(C)C2)C(=O)NC2CCOC2)cc(Br)cc(OC)c1OC C(=O)(C(C)(C)C(C)(F)F)NCC1(CN(C)C(C2(O)CCOCC2)=O)CC1 C1(CC(=O)N(CC(C)NC(=O)CC2CCOC2)C)CCCCC1C N1(C(c2ccc(SCCCC)cc2)=O)CC(NC(=O)C(C)(Cl)Cl)CC1(C)COC c1(OC)ccc(CC(N2CC3CC2C3NC(c2csc(Cl)n2)=O)=O)nc1 N1(NC(CN(C2CC(C#N)C2)C(c2c(C)n[nH]c2C)=O)=O)CCc2nn[nH]c2C1 C(=O)(C1=C(Cl)CC1)N(CCC(=O)NCc1noc(C)n1)CC C1(CC=C)(C(=O)NCC(C)(O)CNC(c2cnc(COC)s2)=O)CCCCC1 c1(C(=O)NCCC2CCCN(C(C(CCC)NC(C)=O)=O)C2)ccc2c(c1)CC2 Cc1cc(Br)ccc1S(=O)(=O)N(c1ccncc1)C(C1CCCCC1)C#N Cc1cc(C(=O)NCCOCC(=O)NC2CC(C=O)C2)ncc1F.N(C)(C)C c1(CCNC(CC(C)NC(=O)COc2ccccc2)=O)cc(O)ncn1 c1(C(=O)NCCN(C(C2CC(C)OCC2)=O)C)cccc(F)c1C(F)(F)F O(N(C)C(=O)CNC(c1ccc(CNC(=O)C#CC2CC2)cn1)=O)CC N1(C(c2cc(C)nn2C)=O)CCN(C(c2cc(F)c(N)cc2F)=O)C(C)CC1C C1(C(=O)NCC2(CN(C(=O)C=CC3CCCN3C)C)CC2)CC(=O)NC(=O)N1 C(CN1C(=O)C(=O)c2ccccc21)(C(C)C)NC(c1cnc(C)s1)=O C[Si](C)(C)c1cccc(NCc2ccc(I)o2)c1 CCC(C)(C)C(c1nnnn1Cc1ccccc1)Nc1ccc(CCCO)cc1 N1(C(C(=O)NCc2c(C)cc(Br)cc2)=O)CCN(C)C(C)C1C C(=O)(C(F)(F)CC(C)C)NCC(CNC(c1c(C)cc[nH]c1=N)=O)C(F)(F)F N(C1CCCc2cc(CNC(=O)C(CC)=CCCC)ccc21)C(C(C)=CC)=O N1(C(C(C(CC)C)O)=O)CC2CCCC2(CNC(C2CCC(N(C)C)CC2)=O)C1 c1(C(=O)Nc2ccc(CNC(C3C=CCC3)=O)cc2)ccc2nccn2c1 C1(CNC(C=NOC)=O)N(C(=O)CCc2cccc(Cl)c2Cl)CCC1(C)C C(=O)(CCCC(=O)N(C)C)NCCC(C)NC1(CS(C)(=O)=O)CC1 c1(NC(C2C(CC=C)C(OC(C)(C)C)C2)=O)cccc2nncn12 Cc1[nH]nc(C(=O)N(CCCNC(=O)CN2CCC(=O)CC2)C2CC2)c1[N+](=O)[O-] CCC(C)C(CN(C)C)NC(C1CC(O)CN1C(=O)CC1CC2C=CC1C2)=O C(CS(=O)(=O)c1cccc(Br)c1)NC(C(CC=C)c1ccccc1)=O c1(COC(c2cn(N(C3(C(N(C)C)C)CC3)CC3(O)CC3)nc2)=O)ccc(F)cc1 C1(NC(CC(CC)C2CCC2)=O)CN(C(=O)CC(CC)CC)CCC1C C1(F)(CNC(C(COC)OC)=O)CCN(C(=O)CCc2ccccc2F)CC1 c1(CC)ccc(C(=O)NC(C)(CSC)C(=O)NCCCc2nc[nH]n2)cn1 N1(C(C(C)(C)CC2CC2)=O)CCCC(NC(=O)Cn2cnc(C#N)n2)CC1 C1(CC(=O)NCC(N(C)C(C2C=CCC2)=O)C2CC2)CCCC(=O)C1 Cc1cc(NC2CS(=O)(=O)CC2NC(=O)C(N2CCC(C)C2)=O)ncc1[N+](=O)[O-] C1(C(=O)NC(C(=O)NCC(COCC)O)C2CC2)CCCSC1C C1(CCC(=O)NCC(COC)C)CCCCN1C(C1CC1(F)Cl)=O C1(C(=O)NC(CC)(COC)CC)CCCCN(C(=O)CCC2CC(C3CC3)C2)C1 CC1C(NC(c2c[nH]nc2F)=O)CCCN1C(c1c[nH]c(=N)nc1C(F)(F)F)=O C1(NC(c2c(C(C)(C)C)ncs2)=O)C2CC(O)C1N(C(=O)C1=CCCCC1)C2 C(CC1CC1)(C(=O)NCCC1(CNC(=O)C(C)CN(C)C)CCCC1)OC C(C(O)C(=O)N1CCC(c2cn(CC3CC4CC4C3)nn2)C1)OC Cc1ccc(C)c(C(=O)NC2CN(C(c3cc(N)cnc3Cl)=O)C(C)(C)C2)n1 c1(CC(=O)N(C2CCCN(C(c3cnnn3CC)=O)C2)CC)n[nH]c(=NC)s1 c1(C(N2CC3C(CNC(CCNC(C4C(C)C4)=O)=O)(C3)C2)=O)cc2c[nH]cnc-2n1 Cc1nc(S)sc1CC(=O)NCC1(CCNC(C23CCCC2CC3)=O)CC1 S(=O)(=O)(c1cc(F)ccc1F)N1CCN(C(c2ccc3scc(C)c3c2)=O)CC1 C(c1cccnc1)=C(C(=O)NCCOCCOCCOCCO)F.C1(CCCC)CCCC1 O=C(C#CC1CCCOC1)NCC1CCN(C(C2CN=C3N=CNN3C2)=O)C1 N1(C(c2ccc(CC)o2)=O)CC23CCCC2(C1)CN(C(=O)Cc1nccn1C)C3 CC1SCCCC1C(=O)NCCOCC(=O)NCc1ncoc1C1CC1 c1(OCCOC)cccc(CN)c1S(=O)(=O)NC(C#N)C(C)CC C1(C(N2CC(CC(C#C)C)C2)=O)C2CC3C(C2NC(=O)C(C2CCOC2)OC)C13 C1(CNC(=O)CC2C3COCC23)(NC(=O)CSC(F)(F)F)CCOCC1 CCC(C(=O)N1CCCC1CN(C)C(c1occc1C)=O)c1ccccc1 C1(C(=O)NCC2CC(C)N(C(c3ccc(CO)s3)=O)C2)CCCC12CCC2 C1(N(C(C(C)N(CCC)C(c2nccs2)=O)=O)C)CC(O)C1(C)C c1(C(C(=O)NCCCF)N(C)CC2(OC)CCOC2)cccc2sccc12 CC1CCCC1NC(=O)NCC1(Cn2nccn2)CC1 C1(C(=O)NCC2N(C(C3CC(OC)C3)=O)CCC2(C)C)CCC2C(C1)C2(F)F C(=O)(C(CCSC)NC(=O)CC1CC2(CCC2)C1)NC(C=C)COC c1(C(N(C)CC2(O)CN(C(C3(O)CC3(C)C)=O)C2)=O)ccc(C2=CCCC2)cc1 C1(CCC)CCOCC1(c1nnnn1C)NCCC(CC)(CC)SC C12(CNC(C(COCC)OC)=O)CCC(CC1)NC2 Nc1cccc(C(N2CC(O)(CNC(c3cn(CC(F)F)cn3)=O)C2)=O)n1 c1(C(=O)NCCCCC2CN(C(CSCC)=O)C2)coc2c1COC2 CCCCC(F)C(=O)NCCC1(O)CN(C(=O)CCC2CCCN2C)C1 N1(C(CCC=C)C)CCCCC1c1cn(-c2cccc(Cl)c2)nn1 C(COC)(CC(=O)N(C(C)CSC)C)NC(c1n(CCC)ncc1)=O c1(C(N2CCC(NC(CCCNC(=O)CO)=O)(CF)C2)=O)ccc(Cl)c(F)c1 N1(C(C(CC=C)(C)C)=O)CC2CCN(Cc3cc(Br)c(F)cc3O)C2C1 CC1CC(CC(=O)Nc2cccc(CSc3ccccc3)c2)C(C)O1 N1(C(c2c(C)noc2C)=O)CCN(C(=O)CC2CC(C3CC3)C2)C(C2CC2)C1 c1(C(N2CCN(Cc3cnc(Cl)cc3Br)C(C(F)(F)F)C2)=O)ccnc(Br)c1F Cc1cc(C(N2CCOC(CNC(=O)C(C3(O)CCCC3)F)C2)=O)cc(O)n1 c1(NCCCC(=O)NC)[nH]c(=NCn2ccnc2)nc2scnc12 C1(NC(C2CCCN(C(C)C)C2)=O)CN(C(C2C(C)C2C)=O)CC1(C)C N1(C(c2nc(NC(C)=O)sc2)=O)CCC2CCN(C(C3CCC(=O)O3)=O)CC12 c1(C(=O)NC2(CNC(C3(C4CC4)CCCO3)=O)CCOC2)cc2ccncc2s1 c1(C(=O)NCc2c(C)noc2C)ccc(-c2ccoc2)c2cc[nH]c12 C1(C(=O)NC(c2ccnc(C)n2)C)(OC)CCCCC1.C12(CC1)CC(=O)NC2 c1(NCC2(O)CCN(C(c3ncccc3C(=O)O)=O)C2)cccc(SC(F)F)c1 C1(CNC(COCC(=C)C)=O)CN(C(=O)Cc2cnccn2)C2(CCOCC2)C1 C(C1CS(=O)(=O)c2ccccc21)NC(c1n(CCCC)nnn1)c1[nH]cnc1C c1(SCC2CCCN(C(c3c(OCC)cccc3)=O)C2)cc(Cl)cc(Cl)c1OC C1(CC)C(NC(=O)CCOCCSC)CCN1C(=O)C(C)O c1(C(C(N2CCC(CN(C)C(C3(O)CC(C)(C)C3)=O)C2)=O)CO)ccc(Cl)cc1 c1(CN(CCOC)CCN2CCc3ccccc3C2)cc2nc(C)cc(C)n2n1 C1(C(=O)NC2(CNC(c3c(C)snn3)=O)CCC2)Cc2ccc(F)cc2C1 C(=O)(N=c1cc(OC)n(C)[nH]1)C1(NC(CC(CCC)CC)=O)CC1C CCCCC(F)C(=O)NC(C1CCN(C(c2cc(CCC)[nH]n2)=O)C1)C N1(C(CCC#C)=O)CCC2(NC(=O)C(F)C3CCC3)CCCCCC12 C1(C(=O)NC(C2CC=CCC2)CC)CCCCCN1C(c1ncc(F)cc1F)=O c12cccc(c1)CNC2=O.CC(C(=O)NCC1CC1C)NC(C)(C)C C1(CN(C)C(c2nc(C3CC3)cs2)=O)CCCCN1C(=O)Cc1ncncc1Cl Cc1ccsc1CC(N1CC(CF)(NC(c2nccn2C(C)C)=O)C1)=O N1(C(CCCCC(C)C)=O)CCCC(C2CN(C(=O)CC3CCC(C)CO3)C2)C1 C1(NC(CCN(CC)CC)=O)CCC(O)CN(C(C2CCCN(C(C)C)C2)=O)C1 C(=O)(C(Cc1ccccc1)N(C)Cc1c[nH]c(C)n1)NC c1(C(CC)Nc2conc2C2CC2)ccc(OC(=O)CC(O)C2CCCC2)cc1 c1(N2CCN(C(C)(C)C)CC2)nc(N2CCNC(=O)CC2)nc(=NCCC#N)[nH]1 c1(OC)ccc(C=NOCC(N2CCCC2)C)cc1.C(C(C)C)N1CCC1.NC c1(CC(N2CCC(NC(CCC=C)=O)C(O)C2)=O)c(C)[nH]c2ccnn2c1=O Cc1cn2c(n1)C(C(=O)NCC(CO)NC(=O)C1CC1)CCC2 C(=O)(C(F)C(C)CNC(C1CC(=O)C12CCC2)=O)NCCC(CCC)C N1(C(C2CCN(C(c3ccc(F)c(C)c3N)=O)CC2)=O)CCC(F)(F)CC1C C1(CNC(C2N(C(COC)=O)CCC2)=O)CCN(c2nnc(C(C)C)o2)C12CC2 N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(F)CC1C(N1CCNC(=O)C1)=O C12(CNC(C(C(C)C)NC=O)=O)CCC(CN(C(=O)C(O)C3CCCC3)C1)C2 c1(NC(N(C(CCCC)C)C)=O)ccc(C(N2CC3CC(O)C3C2)=O)cc1F c1(OS(=O)(=O)Cc2cnn(-n3cc(-c4cccs4)nn3)c2)ccc(CO)cc1 C1(NC(c2ccc(N)cn2)=O)CN(C(=O)CCCC2CC2)C2(CCCC2)C1 n1(CCC(N2CCC(NC(c3c(C)occ3)=O)C2(C)C)=O)cc(S(N)(=O)=O)cn1 c1(C(=O)CN(C(c2cn(CC(F)(F)F)nn2)=O)Cc2ccccc2)ccccc1Cl C1(NC)CCN(C)C(C)C1.Cc1ccc(CN2C(C)(C=O)CC2)s1 CC(=O)CCCC(=O)NCCCCC(C)NC(c1cnnn1-c1ccccc1)=O c1(C(=O)NC2CCCN(C(=O)CCc3cnco3)C2)ccnc2[nH]nnc12 N1(C(C(CNC(=O)C=Cc2ccco2)OC)=O)CC(C)CC(C)(C)C1 C1(C(=O)NCCC(CC)O)CC12CCN(C(=O)COOC1(C)CCC1)CC2 c1(CNCC(c2ccccc2)OC)nc(-c2cnn(C)c2)cs1 C1(C(N2CC(CCCCNC(=O)CCCC(F)F)C2)=O)CCC2(C1)CC2(F)F C(C(C(F)(F)F)n1cncn1)NC(c1cnn(C(F)F)c1)=O.c1(C)ccccc1 C1(C(N2CCCC(NC(c3ccncc3F)=O)CC2)=O)CC12CCCCCC2 C(=O)(CCC(C)C(C(=O)NC(C)C)N1CCC(OC(C)=O)C1)OC N1(C(C(C)C2CC2)=O)CC2COCC(C1)C2NC(c1cn(C2CCC2)nn1)=O c1(C(=O)NCCN(C(CCOCCOC)=O)CC(C)O)c[nH]nc1F C=CCC(CC)C(=O)NC(CCC)CC(=O)NCc1cn(CC)nn1 N1(c2nc(C)c(Br)cn2)CCCC2C1CCN2C(c1ccc2c(Br)cncc2c1)=O C1(CCC)CN(C(C2CC(F)(F)C2)=O)CCN1C(C1COCCN1C)=O c1(C(=O)NC(CC)CN(C(=O)C(c2ccc(Cl)s2)C)CC)cc(C#N)c(C)cn1 C1(CN(C)C(=O)Nc2nc(-c3cnc[nH]3)cs2)CCCN2CCCCC12 C(CC(C(C)C)NC(C1(NC(=O)CC2(CSC)CC2)CCCC1C)=O)OC c1(OCC)ccccc1CCC(=O)N(C(C)CCNC(=O)CP(C)(C)=O)C Cc1cc(CNC(=O)C(C2CC2)N(C)C(C2CCC3(CC3)C2)=O)cc(F)c1 C1(N=c2[nH]nc(C3CC3)s2)(CNC(C2C(C)(CC)C2)=O)CCCC1 CCCCCC(C)CC(=O)N(C)CCNC(C1(C(F)F)CCCO1)=O CC1CN(C(=O)CC2=CCOCC2)CCCN1C(c1cc(Cl)c(F)cc1F)=O CC(CC(=O)NCCOCCCNC(C1(F)CCC1)=O)C1CC1 c1(C(N2CC(C(=O)NC3CCC(C)NC3=O)C(C)C2)=O)ccc2cccnn12 C=CC(C)(C)CC(=O)NCC1CC(NC(=O)CCNc2ccccn2)C1(C)C c1(CC(C)C(=O)N2CC(C)(NC(=O)CCCOC(C)(C)C)C2)ccc(F)cc1F C1(F)(CNC(C2CC=CC2)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1 CCC1=NOC(C(N2CC(O)(CNC(C3CCOC(CC)C3)=O)C2)=O)C1 c1(CCO)cc(C(C)NCCCCOCC(=O)O)cc(Br)c1 C1(CNC(C2CS(=O)(=O)C2)=O)CN(C(=O)CCC2CCCO2)C2CCCC2O1 N1(C(c2ccc(C#C)cn2)=O)CCCN(C(=O)COC2CCOCC2)C(CO)C1 Cc1ccnc(C)c1C(=O)NC1CCCN(C(=O)Cc2cnccc2Cl)C1 C(=O)(C1CCCc2n[nH]cc21)NC1C=CCN(C(c2nc(C)nc(O)c2)=O)C1 CCC(C)(C)C(O)C(=O)N1CCN(C(c2cc(OC)cc(C)c2)=O)C2CCC12 c1(COC)ccc(F)c(NC(c2ccc(C)c(I)c2)=O)c1 c1(C(=O)NCC2CCN(C(c3cc(C(N)=O)oc3)=O)C2)cc(Cl)c(Br)[nH]1 CCC(C)CC(=O)NC(CNC(C1(COCC)CC1)=O)C(C)(C)C C(CCC(=O)NC(c1cccnc1)C(=O)N(C1CCSC1)C)N(C(C)C)C c1(C(=O)NC2C(NC(CCC(C)C)=O)CC2)n[nH]c2ccc(O)cc12 c1(N(CC(=O)NCC2(CC(=O)N(CCN(C(C)=O)C)C)CC2)C)cn(C)nc1C CCCC(F)(F)C(=O)NC1(C(=O)NC2CCC(F)(F)CC2)CCC1 N1(C(C(C)OCCOC)=O)CCCCC1C1(NC(=O)CCNC(=O)COC)CC1 CC(C)(C(=O)NC1CCC(C(=O)NCc2ccncn2)OC1)S(C)(=O)=O C(N=c1[nH]c2cccc(Br)c2o1)C1CCC(NC(Cn2nnc(C(C)(C)C)n2)=O)CC1 c1(-n2c(CC3CCCS3(=O)=O)nc(C(C)OC)n2)ccc(S(=O)(=O)N(C)C)cc1 c1(C(N(C(C(C)O)C(=O)NOCC(F)(F)F)C2CC2)=O)ccn2cncc2c1 C1(NC(CCCCOC)=O)CCC2(CC1)CN(C(c1cc[nH]c(=N)c1)=O)CCO2 N1(C(C(C)OCCCC)=O)CCC(C)C(NC(C2CC3(CSC3)C2)=O)C1 C1(F)(C(=O)NC2CCN(C(CN3C(C)CCC3)=O)CC2)CC2(CCC2)C1 C1(O)(C(CC)C(=O)NCC2(OC)CN(C(c3cnc(S)[nH]3)=O)C2)CCCCC1 CC1(CC(=O)NC2CCCC2CNC(=O)CNC(=O)C2CC2)CCCO1 C1(C(C(N2C(CNC(CN(CC)CC)=O)CC(O)C2)=O)O)CCCCCCC1 C(C)(C(=O)NCCC(C)NC(=O)C(c1ccccc1Cl)C)(C(C)C)OC c1(N(C)C)ccc2ccc(-c3nc(C(=O)Nc4ccc(Br)c(Cl)c4)cs3)cc2c1 c1(C2(C(N(C)CCOCCNC=O)=O)CC(F)C2)ccc(Cl)cc1.c1cscn1 CCC(C)C(C)NC(=O)CCOCCNC(=O)CCc1cnc(C)o1 N1(C(c2c(C)nc(C)[nH]2)=O)CC2CC(NC(=O)Cn3nccn3)C1C2 c1(C(N2CC3C(CNC(CSCC)=O)(C3)C2)=O)c(C)cc(C)nc1Br C(CSC)(C(=O)NCC(C1CCC1)NC(c1sccc1C)=O)OC C(CS(=O)(=O)N(C1CCCC1)CCC#N)(OC)OC C(CCCC)(CC(=O)N(C)Cc1ccn(C)n1)NC(C(CC(=C)C)OC)=O CC(=O)CCCC(C)C(=O)N1CCC(CF)(NC(c2oncc2C)=O)C1 CCCC(CCC)CC(=O)NCCn1cc(C(=O)NC2CCN(CCC)C2)nn1 c1(OC)cc(F)c(C(N2CCC(NC(=O)C3=CCC3)CC2C2CC2)=O)cc1OC c1(CC(N2CC(C(C)NC(c3csnc3Cl)=O)OCC2)=O)cc2ccccc2s1 c1(C(=O)NC2CCCC(Nc3nc(SC)c(C)cn3)C2)ccc(P(C)(C)=O)o1 c1(C(=O)NCC23C(CN(C(C=Cc4n(CC)ccn4)=O)C2)C3)c(C)ccnc1C CC(CO)CCNC(=O)NCC=CCNc1cc(C2CC2)no1 c1(CC)ccc(C)c(C(=O)NC(CCNC(c2cnn[nH]2)=O)C(C)C)c1 CC1(C)CC(C(=O)Nc2cc3c[nH]cnc-3n2)CN(c2nc(C#N)c(Cl)s2)C1 N1(C(C=CC)=O)CC2(CCC2NC(C2CC(=O)NC(=O)N2)=O)C1 N1(C(C(n2ccc(C)n2)C)=O)CC2CC1CN2C(=O)Cn1cnnc1 C1(C(=O)OC)(NC(CCC#C)C)CC2(CCCCC2)C1 N1(C(c2c(CC)nc[nH]2)=O)CCC(N(CC(C)C)C(c2cc[nH]c2)=O)CC1 c1(C(=O)NC(C2N(C(C(CC=C)C)=O)CCC2)C)[nH]c2cc(OC)ccc2c1C N1(C(C2(C=C)CCC2)=O)CCC(NC(=O)Cc2c(F)cccc2F)C(CO)C1 CC1(C)C(C)(C(=O)NCCCNC(c2cc(N)nc(Cl)c2)=O)C1(C)C N1(C(CC2(COC)CC2)=O)CC(NC(=O)CC2CC(OC)C2)C(C)(C)C1 N1(C(CSCC=C)=O)CC(N)C2(CC2)C1.C12CCN(C1)C(=O)COCCOC2.CC N1(C(c2c(Cl)ncc(N)c2)=O)CC(CNC(c2nocc2Cl)=O)OC2COCC12 c1(NC2CCCCN(C(C3(C(C)C)COC3)=O)C2)ncnc2sccc12 C1(CC(=O)NCc2nc(C)on2)CCCN(C(=O)C(CCN(C)C)N(C)C)CC1 Nc1sc2ccccc2c1C(=O)NCC1CCCN(C(=O)C=Cc2cnc[nH]2)C1 c1(C(=O)NC(c2cc(Br)cs2)C2CCOC2)cn(C)nn1.CC1CN1 N1(C(=O)Nc2ccnn2Cc2noc(C3CC3)n2)C2CCCC1CC(O)C2 C(=O)(C(C)(C)CO)N(CCC(C)NC(=O)COC(c1nccn1C)C)C c1(C(=O)NCC(C)NC(C2C(C)CC2)=O)ccnc(C2CCCC2)n1 CCCCC(CC)C(=O)N(C1CCN(C(=O)CC2CC(=O)C2)C1)CCO C1(NC(C(C)C)=O)CC2CCC1N(C(c1cc(F)n[nH]1)=O)C2 C(c1ccc(Cl)c(Cl)c1)=CC(=O)N(CC(CNC(C1ON=C(C)C1)=O)(C)C)C C1(NC(C2N(C(c3c(CC)n(C)nc3)=O)C(C)C2)=O)CCC2(CCC2)C1 N1(C(c2c(OC)cncc2)=O)CCOCCC1C(N1CCOC(C)(C(N)=O)C1)=O c1(CC)ccnc(C(N2C(C(=O)NCCc3nccnc3C)CCC2CC)=O)c1 C(=O)(CCCC(C)NC(=O)C(C)SC)NC.C12(CCCCC1)C(=O)N2 C(=O)(CCN(OC)C(=O)CNS(C)(=O)=O)N1C(C#C)CCCC1 C12(C(N(C3CN(Cc4ccc[nH]4)CC3O)C)=O)CCC(CC1)C2 c1(C(=O)NCC2(NC(C3CC(=O)NCC3)=O)CCOC2)ccc2c(c1)CCCS2 N1(C(=O)CC2(CNC(=O)C3CC3)CC2)CCOCC1=O.c1(N)cc(C2CCOC2)on1 C1(CNC(C2CC(CCNC(c3oc(C)c(CO)c3)=O)C2)=O)CC2CCC1CC2 CC1CCC(NC(=O)C(F)(F)C2C(N)CCC2)CN1Cc1ccccc1 C1(NC(CCN(CC)CC)=O)CC2CCC1CN2C(=O)Cc1ccns1 CCCC(C(=O)N1CCC(C(=O)NC(C)CF)C1)C(C)C c1(NS(C2(CCC=C)CC2)(=O)=O)c(C)ccc2cccnc12 C(=O)(CS(=O)(=O)C(C)C)NC1CCN(C(c2c(C)cccc2C)=O)C1 C1(NC(c2n(CCC)ncc2)=O)CC2CCC1N2C(=O)C=Cc1ccc(F)cc1 c1(-n2c(-c3ccc(-c4ccccc4)o3)nc(C(C)O)n2)ccc(CO)c(Br)c1 c1(CC(C(N2CCC(N(C(C(C)=O)=O)CCO)C2)=O)C)cccc(F)c1 C1(NC(C=CC)=O)CC2CCC(C1C)N2C(=O)C(c1ccnn1C)OC Cc1ccc(CCCNC(c2nnnn2CSC(C)CCc2ccco2)C2CCC2)o1 C(=O)(C1=CC2C=CC1C2)N1C(C)C(C(=O)NCC2(CCCO)CC2)CC1 N1(C(c2cc(C(CC)C)no2)=O)CCC(NC(=O)CCSCC(N)=O)C1C(C)C c1(CN(C(c2ccn(CC(F)(F)F)n2)C(=O)NCC(=C)C)C)cccc(Cl)c1 Cc1cc(Br)cc2[nH]c(C(=O)NC(C)CN(C(=O)CN(C(=O)COC)C)C)cc12 C=CC1(NC(=O)CC2CCCN2C(c2[nH]ccc2C)=O)CCCC1 c1(NCCSc2n(C)ncc2S(N)(=O)=O)[nH]c(=NC2CC2C)nc2c1cnn2C Cc1ccc(O)c(NC(=O)CC(CC2CC2)NC(=O)C(CO)NC(N)=O)c1 N1(C(CC(C)OC)=O)CC2(NC(=O)CC(CC)C3CC3)CC1C2.c1(S)ccccc1Cl C1(C(=O)NCCS(=O)(=O)CC)(NCc2ncsc2C)CCCC1C C(=O)(CCS(=O)(=O)Cc1ccccc1)N1CCCC(N(C)C2CC2)C1 N1(C(=O)CCN2CCCC2)CCC(O)(Cc2cn(-c3cccc(Br)c3)nn2)CC1 C1(N(C(c2cccc(SC)c2)=O)C)CCCN(C(=O)C(C)CSC(F)(F)F)CC1 N1(C(c2c(OC)nsc2)=O)CC2(NC(c3coc(Cl)n3)=O)CC1C2 N1(C(C2(OCC)CCCC2)=O)CCC(C(C)NC(C2(C(C)(F)F)CCC2)=O)CC1 C1(CNC(=O)C=CC=C(Cl)Cl)CC2(CC2)CN1C(=O)CC1CC(C(F)F)C1 CCCCC(CC)C(=O)NC(CCCNC(=O)C=C(C)C(C)C)c1ccccc1 C(=O)(C#CC1CCCCC1)NC1(COC)CCN(C(=O)CCCn2cncn2)C1 c1(C(N2CCC(C(C)C(=O)NCCC(O)CO)C2)=O)ncccc1O N1(C(c2cc(C(C)C)on2)C(=O)NCC=C)CCN(CC2CC2)CC1 CC(C)CC(C)(C(N)=O)NC(C1CC(NC(C2SCCS2)=O)C1)=O Cc1ccc2c(c1)N(C(=O)C(N1CCc3ccccc3C1)=O)CC2 c1(OC)cc(OC)c(Cl)c(C(=O)N(CC(C2CC2)N(C)C)C)c1 c1(CNC(N2CCN(C3CC3)C(=O)C2)=O)nc2cccnc2[nH]1 c1(C(N2C(CCC(N3CCCC(OC)C3)=O)CCC2)=O)ccc(O)c(Cl)c1 C12(C(=O)NC3CC(CN=[N+]=[N-])C3)CCC(CN(C(C3CC4C=CC3O4)=O)C1)C2 Cc1[nH]c(C(N2CCC(C)C(NC(=O)CS(=O)(=O)C(C)C)C2)=O)c(C)c1C N1(C(COCCC#C)=O)CCC(C(C)NC(c2ccn(C(CC)CC)n2)=O)C1 O=C(C1=Cc2ccccc2OC1C(F)(F)F)Nc1ccc2n[nH]cc2c1 C1(CNC(C(N)=O)=O)CCN(C(c2cccc(C(N)=O)c2)=O)CC1O CC(Cc1ccco1)N=c1cccc(S(=O)(=O)N2CCSC2C(F)(F)F)[nH]1 CN1CCC(N(C=O)Cc2c(Br)n[nH]c2Br)C1=O C#CC1(C(=O)NC(C)CC(C)CC)CCN(C(c2cnc(OC)s2)=O)CC1 C1(C(=O)NCCC(C)F)CCCCN(C(C2C(C)(C)C2(F)F)=O)C1 C1(CNC(C(C)NC(=O)OC)=O)CN(C(=O)CCCC(N)=O)CCC1C CN1CC2(CCCN(C(CCCC3CC3)C(=O)NC3COC3)C2)CC1=O C(=O)(CCCCO)NC1(c2ccccc2)CCC1.C12CCN(C1)C(=O)N(C)C2 C(CC(CCCC)C(=O)OC)NC(=O)NC(c1ccccc1)CC=C c1(OC)ccc(C)nc1C(N1CCC(N(C(=O)C(C)n2ccnn2)C)CC1)=O C(=O)(C(C1=CCCCCC1)N1CCOC(C2CCC2)C1)NCCC c1(CC)noc2ncc(C(N3CC(NC(=O)CCF)CC(O)C3)=O)cc12 CCCC(C(=O)N1CCCC1C1(NC(C2CC2OC)=O)CC1)N(C)C C1(C(=O)NCC(O)C2CCC2)(SC)CN(C(=O)Cn2ccc(C)n2)C1 c1(C(N2CC(CNC(c3cc4scnc4[nH]3)=O)OCC2)=O)cccc(Cl)c1O Cc1cc(=NCc2nc(C3CCCO3)n[nH]2)[nH]c(N(C)CCN2CCN(C)CC2)n1 c1(CC(=O)NC(C2CCCCC2)CNC(C(CC)SC)=O)c(F)cccc1F c1(N(C(C(F)=CCC)=O)CC(N2CC[Si](C)(C)C2)=O)ccc(F)c(F)c1 C1(C)(C(=O)NC2C(N(C)C(=O)C3CC3c3ccccc3)CCC2)COCC1(F)F C(=O)(C(F)(F)CC(C)C)NCC1(C)CCCN(C(C2(CC#C)CC=CCC2)=O)C1 N1(C(C2(CC=C)CC2)=O)CCC(NC(c2cnc(N)c(Cl)c2)=O)C(C(C)C)C1 CC#CC(c1ccccc1)=CC(=O)NCC1CCCCN1c1cc(C)nc(SC)n1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(CC=C)(NC(C(C=C)O)=O)C1 NC(COc1ccccc1)CC(=O)N1CCN(c2cnsn2)CC1 c1(C(N2CC(NC(c3nccc(C)n3)=O)C3(C2)CC3)=O)ccnc2[nH]c(C)nc12 CC(C(=O)NC1CCCCC1NC(c1cncnc1)=O)S(=O)(=O)C1CCOCC1 Cc1c(C(N2CC(NC(C3CC3C(C)C)=O)CC(F)C2)=O)nn2c1CCCC2 CC1(C(F)F)CN(C(C(=O)NC2CCCCC2)c2nc[nH]n2)CCO1 C1(C(=O)NCC(CNC(CC2(CC)CCC2)=O)C(F)(F)F)CCn2ncnc2C1 C#CC1(C(N2CCC2(C)CC(=O)NCC2(C)CCCC2)=O)CCCCC1 N1(Cc2cccc(CC#N)c2)CCC2(CCN(S(=O)(=O)CCBr)C2)C1 c1(CC(=O)NC2(C)CN(C(COC3C(C)CCCC3)=O)C2)cnc2n1CCOC2 c1(C(=O)NCC(CNC(c2c(CC)noc2C)=O)C)c[nH]c2cc(Cl)ccc12 N1(C(C2(COC)CCN(C(c3sc(C)nc3C)=O)C2)=O)CCSCCC1C c1(C(=O)NC(C(C)NC(c2n(CC)nc(C3CC3)c2)=O)C)cc2ccccc2[nH]1 CC1Cc2c(Br)cccc2CN1C(=O)NC1CC2(C1)CC(O)C2 N1(C(c2c(C(C)C)con2)=O)CC(N(C)C(c2ncc(F)cn2)=O)C(O)C1 CC1(C)C(NC(=O)CC2CC(F)C2)C2CCCN(C(C3COC4COCC34)=O)C12 N1(C(CN(C(CC(C=C)C)=O)C2CC2)=O)Cc2cccc(C#N)c2C1 c1(C(=O)NCCN(C)C(c2cnn[nH]2)=O)cccc(C2CC(F)(F)C2)c1 N1(C(c2cc(CC)no2)=O)CC(NC(c2ncccc2F)=O)C(n2ccnn2)C1 c1(C(C)=O)ccc(CC(N2CCC(C)(NC(C3CCC3C(F)F)=O)C2)=O)cc1 C(CN=c1nc(N2CCC(C(F)(F)F)C(C)(C)C2)c2c([nH]1)CCC(C)C2)SC C1(CC(=O)NCC2N(C(C(C)NS(CCC)(=O)=O)=O)CC2)CCCNC(=O)C1 c1(-n2ccc(C(N3CC(N(C(C(C)CF)=O)C)C(F)C3)=O)n2)ccc(F)c(F)c1 C1(NC(C(COC)C)=O)CCCCC12CCCN(c1ncc([N+](=O)[O-])cc1Cl)C2 c1(C(=O)NCC(C(C)C)NC(CC)COC)ccc2ccoc2c1 c1(C(N(CC(CC)OC)C)=O)cc(CNC(=O)CC2(CO)CC2)ccn1 c1(C(=O)NC2(C(=O)NCc3nnc(C)o3)CC(F)C2)ccnc2cc[nH]c12 C1(C)(NC(C(C)(C2CCC2)NC(CC(C=C)(C)C)=O)=O)CCCCC1(C)C N1(S(CC=Cc2cncc(C)c2)(=O)=O)CC2CCC1CN2C(=O)NC1CC1 C12(C(=O)NC(c3nccs3)C)COCC1CN(C(C1CCCC(CF)C1)=O)C2 c1(C(N2CCN(C(C(C3CC3)OC)=O)C(CF)C2)=O)cnc2ccc(F)cc2c1 C1(C2(O)CCOCC2)(NC(C2CCCN2Cc2ccccc2Cl)=O)CC1 C1(CCC(=O)NCCCSC)CCN(C(=O)C(C)(C)OCC=C)CC1 n1(C(C(=O)NC(CC)CNC(c2cc3ccsc3[nH]2)=O)C)cnc2ccccc12 Cc1cc(C(=O)N(C(C)CCNC(C2(CC(F)(F)F)CC2)=O)C)c(C)[nH]1 C1(CC(=O)NCCC2CCN(C(CC(C)(C)C#N)=O)C2)CCC2(CCCC2)CC1 Cc1ccc(OCCC(N2CCCC(CCNC(C3COC(=O)N3)=O)C2)=O)cc1 C1(C(=O)NCCSC)CCC2(CC2)N1C(c1csc(O)n1)=O CCC(C)C(C)C(=O)N(CCCNC(=O)C=Cc1cn(C)nn1)C N1(C(CN(C)CC)=O)CCN(C(c2ncc(Cl)cc2O)=O)CC1c1ccncc1 C1(NC(C(C)SCCCC)=O)CN(C(c2nnn(C)c2C)=O)CCC1(C)C N1(C(C2(CC#C)CC2)=O)CCCC(O)(CCNC(c2ccc(C)cc2F)=O)C1 N1(C(c2c(C)ccc(C)c2)=O)CC2(CCCC2NC(=O)CN2CCN(C)CC2)C1 c1(C(=O)NCC2N(C(Cc3ccc(OC)cc3F)=O)CC2)cc(Cl)c(F)cc1O C1(CNC(C2C3COCC23)=O)CCC(C(N2CCCC(CC3CC3)C2)=O)CC1 c1(C(N2CC(C)(NC(C(C)Cc3ccncc3)=O)C2)=O)cc([N+](=O)[O-])ccc1O Cc1nn(-c2ccc(Cl)cc2)c(Cl)c1CNc1cnc(CN2CCOCC2)s1 n1(CCCC(=O)NCCOCCCN(C(C(C)CC2CC2)=O)C)cnc(C#N)n1 N1(CCC(N2CCC(C(=O)Nc3c(C)nsc3)C2)=O)CCc2ccccc2C1 c1(C(N2CCCC(CNC(C(C=C)(C)C)=O)C2)=O)c(C)nn(CC)c1Cl CCCCCCCCC(=O)NC(CC(C)(C)C)C(=O)Nc1cccc([N+](=O)[O-])c1 c1(-c2cc(OCOC)cc(F)c2)cc(C(=O)NCC#N)cc2[nH]ncc12 CCCCC(CO)NC(=O)CN(C(=O)CCc1cncs1)CC c1(C(N2C(C)CN(C(C3(Cl)CC3(F)F)=O)CC2)=O)ccc2c(c1)COCO2 CCCC(O)C(CO)NC(=O)C(C)CCCc1ccccc1 c1(C(=O)NC2CC(N(C(c3cc(CC)cc(N)c3)=O)C)C2)ccc(F)c(C)c1Cl c1(CN(CCC(F)(F)F)C(C2N(C(C)=O)CC(O)C2)=O)ccc(Cl)cc1Cl C1C(=O)N2CCC(O2)C(=O)N1CC.C1(SCC)C(C(C)=O)C1(C)C.C(=O)OC CCCCCCN(CC)C(C1COC(C)C1)=O.C1(=O)CCN1.[SH](C)(=O)=O C(=O)(C(C)C(C)COC)N1C(N(CCc2ccc(OC)cc2)C)CCCC1 N1(C(C2CC(=C)C2)=O)CCC2(CCCN2C(C2(c3ccno3)CCC2)=O)C1 N1(C(c2cc(CC)n(C)n2)=O)CCN(C(c2nccc(C(F)(F)F)n2)=O)C(C)C1 C1(NC(=O)C=C2CCOCC2)CCCC(CNC(=O)CCn2cnnn2)C1 CP(C)(=O)CC(=O)N1CC(O)(Cc2nnnn2-c2ccccc2)C1.C1(=O)NO1 c1(C(=O)NCC2CCN(C(COCP(C)(C)=O)=O)C2)ccc2n[nH]cc2n1 c1(NC(=O)CCC2CCN(C(c3ccc(O)c(F)c3)=O)C2)cccc(F)c1F C12(CN(Cc3cc(C)oc3C)Cc3ccccc3C)CCCC1CCO2 N1(C(C(n2c(C)ncc2)C)=O)CCCC(NC(=O)CCc2nc[nH]n2)C1 N1(C(c2ncc(NC)nc2)=O)CCCC12CCN(C(=O)C1=CC(C)(C)C1)C2 CC12CCC(CC1)N2.C1(NCc2ccccc2)CCCN(O)C1=O c1(C(N2CCN(C(c3c(C)nco3)=O)C(C)C2)=O)ncc2[nH]ncc2n1 CC1(C)CC(CNC(c2ccc[n+]([O-])c2)=O)N(C(c2ncc(C(F)F)s2)=O)C1 c1(-c2cn(CC(=O)N(C)CC3CC(c4ccccc4)CO3)nn2)ccc(Cl)cn1 C1(NC(CC2(N(C(C(CC)(C)CO)=O)C)CC2)=O)CCC([N+](=O)[O-])CC1 Cc1nc(Cc2cn(C(C(F)(F)F)c3ccccc3)nn2)no1 Cc1[nH]nc2ccc(C(=O)NC(C3CCN(C(c4cc(N)ccn4)=O)C3)C)cc12 c1(C(=O)NCC2CC2OCCCNC(CCSCCOC)=O)cn(C2CC2)nn1 N1(C(C(C)NC(=O)Cn2cnnn2)=O)CCN(c2nc(C(F)(F)F)ns2)CC(O)C1 C=CC1(CC(=O)NC(C)(CNC(=O)C=CC(C)C)C2CCC2)CCC1 N1(C(c2nnn(CC)c2C)=O)CCCCC12CNC2 O=C(CC1CCN(C(=O)Cc2cc(O)cc(F)c2)C1)N=c1ccn(CCO)[nH]1 c1(OC)nc(C(=O)NC2CCC2C(=O)N(C)Cc2ncc[nH]2)co1 C(C(=O)NCCOC(CC(=O)NC(C)(C)C)C(C)C)(C(C)(C)C)SC C1(CCOCC)CCN(c2nnc(C(N3CCOC(CC(=O)OC)C3)=O)s2)CC1 C1(NC(c2cccc(F)c2)=O)CN(C(=O)C(F)Cc2ccccc2)C2(CCC2)C1 C12(CCNC(=O)CC3CCC4CC34)CC3CC(CC(C3)C1)C2 CCC(CC)C(C)C(=O)NCC1(C)CN(C(c2ccnc(OC)c2)=O)CCO1 C1(CC)CCC(C)CN1C(c1ccc(C(F)(F)F)o1)C(=O)NCC1CCOC1 C12(C(=O)NC(CC#C)(C)C)CC1CN(C(c1cccn1CC#C)=O)C2 C(=O)(CS(=O)(=O)C(C)(C)C)N1C(CN(C(C=C2CCC(C)C2)=O)C)CCCC1 C1(C(=O)NC(C(=O)N(CCS(C)(=O)=O)C)C2(C)CC2)CCCC(=O)N1C CCCC(C)CC(=O)NC1(C)CCN(C(C2(C(F)F)CCCCC2)=O)C1 C1(C(N2CC3(CN(C(c4ccn(C(C)CC)c4C)=O)C3)C2)=O)CCOCC12CCC2 C1(CCC(=O)NCc2[nH]c(=N)sc2)CCN(C(C2C3CCC(F)C23)=O)CC1 c1(C(=O)NCC2(OC)CCN(C(c3c(C)cnn3C)=O)C2)ccc(S(C)=O)cc1 c1(-c2cn(C3CCC(C(=O)NCCc4ccc(C)s4)C3)nn2)ccc(O)cc1Cl c1(C(C(=O)OC)NC(=O)C(C)NCC(C)(C)C)ccc(OC(F)F)cc1 c1(CCC)cccc(C(=O)NCC2CN(C(=O)C(C)Cc3cnc[nH]3)CCO2)c1 c1(C(=O)NC(CCNC(C(C2CC(F)(F)C2)OCC)=O)C)cc(Cl)ccc1C N1(c2nc(Cl)nc(CC)c2Cl)CC23CCCC2(CN(C(C2CC(C)=NO2)=O)C3)C1 c1(C(=O)NCC2CC(C)N(C(c3ncc(F)cc3F)=O)C2)ccc(F)c(O)c1 C1(C(=O)NCC2(NC(C=CC(C)C)=O)CCCCC2)C2CCC1(C)C2(C)C C(=O)(C(C)(CC)CO)N(CCC)CCNC(c1cncc(F)c1Cl)=O C1(c2nnnn2C2CCOC2)(NCCCc2ccncc2)CCC2(CC1)CSC2 N1(C(C(C)N(C(C2(C)CCCC2O)=O)C2CC2)=O)CC(CO)CC(C)(C)C1 C(=O)(CC(C)(C)CNC(c1cc(CCO)on1)=O)NC(CN(C)C)CO N1(C(C2N(C)CC2)=O)CC(F)(C(F)C(=O)O)C1.C1(C(=O)OC(C)(C)C)CNC1 C(N=c1ccc(Br)c(S(=O)(=O)NC2CCc3nccn3C2)[nH]1)C1(C)CC2(CC2)C1 C(=O)(C(F)CC(C)(C)NC(C1OCC2CCCC12)=O)NC(c1cccs1)C C(=O)(C(O)CC(F)(F)F)NCC1(C(=O)NC2CC(C)C2)CCCC1 C1(C(=O)NC(CC2CN(C(C3CC(=C)C3)=O)C2)C)CCCN1C1CCCC1 C1(CNC(CCOC)=O)CC2(CCN(C(C3C=CC=CC=C3)=O)CC2)C1 C1(CNC(C(C)NC(c2ccoc2)=O)=O)(CO)CCN(C(=O)CC2CC23CC3)C1 N1(C(=O)CC2CC=CCC2)CCN(C(=O)CN2CCOCC2)C(C2CC2)C1 c1(C(=O)NC2C(NC(CC3CC(C)(C)OC3)=O)C2)c(Br)ccc(F)c1N C1(CNC(=O)CCCc2ccsc2)CC2CCC(C1)N2C(=O)Cn1cccn1 CC1(C)CCC(n2cc(C3CC3CO)nn2)CN1C(c1ccc2nsnc2c1)=O C(c1ccccc1)=C.C(=O)(C(C)OCCN(C)C)NCC(C)NC(=O)CO C1(CCOC)(C(=O)O)CC2CC1C2.C1CC(=O)N1 c1(OC)cnc2[nH]c(C(N3CCC(NC(C4(C#N)CCOCC4)=O)C3)=O)cc2c1 Cn1cc(CCNC(=O)CC2CCN2C(C2CC(F)(CF)C2)=O)nn1 C1(CC(=O)NCC(C)(C)N(C)C)CC=CCC1.C1(=O)CCN1C.C(CCO)N CC1(C)CC(C(=O)NCc2ccnc(C#N)c2)N(C(C2CC2C(N)=O)=O)C1 CC1(C(=O)NCc2ccc(C(=O)O)s2)CCc2ccccc21 C1(C(N2CC3C(CNC(CSCC)=O)C3C2)=O)(COC)CCCNS1(=O)=O N1(C(C(C)SCC)=O)CCCN(C(=O)C(c2cc(F)cc(F)c2)O)CCC1 C1(CNC(C2(C)CCNC2=O)=O)CCC2(CN(C(c3ncc(F)cc3F)=O)C2)O1 n1(CC=C)cc(CC2CCCN2C(c2cc(CCC)[nH]n2)=O)nn1 c1(NC(C2CC2CNC(=O)CC23COC(CF)(C2)C3)=O)cc(O)ncc1C(F)(F)F N(C(=NCCF)NCc1ccccc1C)OC.C1CCC(OC)(OC)C1 C1(CC(=O)N(C)CC2(NC(C3CC(=O)N(C(C)C)C3)=O)CC2)CCCCC(=O)N1 c1(C(=O)NCC2C(NC(c3cnn(C(F)F)c3)=O)CCC2)ccncc1Cl C1(N(C)C(c2cocn2)=O)CC(NC(=O)CC2CN3CCC2CC3)C12CCC2 c1(CNC(c2n(CCCSC)nnn2)C2CCCCC2)cccc(Cl)c1Br c1(CNC(c2ccc(C)cc2)CCOC)ccc(-c2cnn(C)c2)cc1F CC1=C(C(=O)N2CCN(C(c3cc(C(C)C)[nH]n3)=O)CC2CO)S(=O)(=O)CCO1 Cc1c(C(=O)NC(C)(C)C(C)NC(=O)C2=NN(C)C(=O)CC2)oc2ccccc12 C(C)(CCCCNC(c1ccc(C(C)C)cn1)=O)NC(CSC)=O c1(C2(C(N(C(CNC(C3(N(C)C)CC3)=O)C3CC3)C)=O)CCC2)ccccc1C#N c1(C(=O)NCC2(F)CCN(C(c3ccsn3)=O)C2)cccc(-c2cncnc2)c1 N1(C(c2cc(OC)ncc2Br)C(=O)NC2COC2)CCC(O)(C#CBr)CC1 C1(NC(c2cc(COC)on2)=O)CN(C(=O)CSc2nncs2)CC2CC12 c1(C(=O)NCCCC(C)NC(c2conc2C2CCCO2)=O)cccnc1S Cc1csc2ccc(-c3ccnn3C(F)(F)F)cc12 c1(C(N(CC(CC)NC(=O)C(N2CCC(C)CC2)=O)C)=O)cncc2ccsc12 C(C)(C(=O)NC1CC1C(=O)NC1CN(C2CCC2)C1)SC C1(NC(c2c(C)nc(CC(C)C)s2)=O)CCCCN(Cc2cscn2)C1 CC1C(=O)CCC1C(=O)NCC1CC(C(=O)NC(c2nnnn2C)C)C1 c1(OC)cccc(CC(=O)NCC(C)CNC(=O)C(C)NC(C)=O)n1 C1(COC)(CNC(=O)CC2CC2)CCN(C(C2(Cl)CC2)=O)C1 c1(C(=O)NCCC2CCCN(C(C(CC(=C)C)C)=O)C2)ccsc1S(C)(=O)=O N1(C(C(c2ccccc2)C)=O)CC(CN(C)C)CC(C)(C)C1 CCC(CNC(=O)Cn1nccc1C)(CC)C(=O)N(C1CCOC1)C c1(C(N(C)C)=O)cncc(C(=O)N(C2CC(NC(=O)CN(C3CCC3)C)C2)C)c1 CP(C)(=O)C(O)C(=O)N1CCC(O)(CCNC(c2cnoc2C2CC2)=O)CC1 C(C(C)(O)CNC(c1cn(C(C)C)nn1)=O)NC(C1C(COC)C1)=O c1(NC(=O)Nc2ccc(C(N3CCOC(C(F)(F)F)C3)=O)nc2)cccc(O)c1 Cc1c(NC(c2ccc(OCCO)cc2)C)ncnc1NCC1CNC(=O)CO1 N1(C(c2ncc(OCC)s2)=O)CCCC12CCN(C(=O)C(C)CC1CCC1)CC2 N1(C(C(CC2CC2)NC(C=C(CCC)CCC)=O)=O)CCCOC(C)C1 CN1CCN(C(C2(CO)CCCO2)=O)C(CNC(=O)CN2C(=O)CCCC2=O)C1 c1(C(=O)OCc2scc(C)n2)ccc(F)c(Cl)c1.N12CCCC1C2=O C(CC(C)C)(C(=O)NC1CCCCC1NC(C)=O)N(CCCC#C)C C1(NC(C(=O)N(CCC)CC2CC(F)(F)C2)=O)CS(=O)(=O)CC1OC c1(N2CCCC(NC(=O)C(F)C3CCOC3)C2)ncnc2[nH]ccc12 CCCN=C(NCC1CCCN1C(=O)OC(C)(C)C)NCC1C=CC2CC1CO2 c1(C(N2CC3CC(CN(C(C=CC)=O)C3)C2)=O)cc(S(C)(=O)=O)ncc1Br C1(C(=O)NC2CCC(OC)C2)CC2CC1CN(C(c1csc(=N)[nH]1)=O)C2 C#CC1CC2(CC2)CN1C(=O)CC(CNC(c1cc(C(C)=O)[nH]n1)=O)OC c1(CC)ccc(F)c(C(N2CCC(NC(=O)COCc3ccncc3)C2C)=O)c1 c1(CC(=O)N(C2CCN(C(=O)CCCOC(C)(C)C)C2)C)ccnnc1O S(=O)(=O)(c1ccc(C(N)=O)cc1)NCC(=O)NC(C(C(C)C)O)C C1(C2CC2)(C(=O)NCc2cn(C3CCN(C(C=CCN(C)C)=O)C3)nn2)CCC1 N1(C(CNC(N)=O)=O)CCN(C(=O)Nc2cc(F)cc(F)c2)CC1CCO C1(CNC(C(C)=CC2CC2)=O)C=CCN1C(=O)C(C)OCC1CCCCO1 C1(C)(C(=O)NC(CN(C(=O)Cc2cn[nH]c2)CC)C)CCCN(C(C)=O)C1 C(=O)(C(CC(C)C)C(C)C)N(CC(C)NC(=O)CC(N)=O)CC c1(-n2c(-c3c(F)nc(Cn4cnnc4)[nH]3)ccn2)ccc2nncn2n1 C1(NC(=O)COC2CC(F)(F)C2)CN(C(C2CN3CCC2CC3)=O)CC2CC12 C1(CCC(=O)NC(CNC(CCN(CCCCOC)C)=O)CO)CCCCCC1 c1(C(N2CC(NC(c3nc(OC)oc3)=O)(CO)C2)=O)cccnc1C(F)(F)F C1(CNC(Cc2c(C)non2)=O)CC2CCCC2N1C(=O)C(F)C1CCCC1 C(CC(O)C(=O)N(C)CC1CCC(=O)N1)NC(COC1(C#C)COC1)=O C(=O)(CCCCNC(N)=O)N1CC(CC=C)(NC(=O)NCCCC(=O)NC)C1 c1(C(=O)NC2C(NC(c3ccnc(CO)c3)=O)CCC2)cnc2sccn12 N1(C(C(CC2CC2)OC)=O)CC(C(=O)N(C)C(c2ncccn2)C)CC(C)(C)C1 C1(NC(c2occ(C)c2)=O)C2CC1CN(C(=O)CCOc1ccccc1F)C2 N1(C(C2(C#N)CC3(CC3)C2)=O)CC2CCCC2(CNC(=O)CO)C1 C1(N(C(=O)CC(CC)C2CCC2)C2CCN(CC)CC2)C2CCOC2C12CCCC2 C(=O)(N=c1[nH][nH]c(C)c1Cl)C1C(NC(c2c(C)nc[nH]2)=O)CCC1 C(CCC(=O)NCC1COC(Cc2nncn2C)C1)SCCOC.C1(=O)C(C)N1 N1(C(c2cc(OCCCCC)no2)=O)CC(F)(F)CC1C(=O)OC(C)=O Cc1ccc(C(=O)NCC2(O)CCN(C(C3CCC(C)(C)C3C)=O)CC2)c(C)c1 C1(OCC)CCN(C(=O)OC(C)(C)C)CC1C.C1(=O)CC(C)(C)N1 c1(CNC(C#CCN(CC)CC)=O)ccc(Cl)cc1C(F)(F)F CCC(CCC(=O)Nc1ccc(C)c(C)c1)NC(C1CN(CC)CC1C)=O C1(C)(C(N2CC3C(CC(NOCC(CC)C)=O)C3C2)=O)CCN(C)CC1 CCC(C)(C)C(=O)NCC1(NC(=O)CC2COCC2(C)C)CCC1 c1(C(=O)NC2CC(NC(c3ccsn3)=O)CC2O)c[nH]c2nc(Cl)ccc12 C1(CNC(CCCCOCC)=O)CN(C(c2c[nH]cc2C2CC2)=O)CC(C)(C)O1 c1(Nc2ccc(N3CCC(=S)NC3=O)cc2)ccnc2c1ccc1ccccc21 N1(C(c2cc(CCC)oc2C)=O)CCC2(CCN(C(=O)CC3CCSCC3)C2)C1 C1(C(=O)NC2CCN(C(C3CC4=C(C3)N=N4)=O)C2)CC2C=CC1CCC2 c12ccc(c(F)c1)[nH]c2=O.C1(C)(C(=O)NCc2cn(C)nc2)CCCN1C(C)=O C1(NC(N(C2CCN(C)C2)CCC)=O)CCCN1Cc1ccccc1 C1(OC)CCCC(CC(=O)NC(C2CCCCC2)C(=O)NC2(C)CCCC2O)C1 N1(C(c2c(CCOC)ocn2)=O)CC2(CCOCC2)CC1CNC(=O)C(C)SC N1(C(CC(C(=C)C)OCC)=O)CCC(C#CC)CC1.N12CC(C1)OCC2 C1(C(C)NC(C2CC2CC(C)(C)C)=O)CCN(C(c2cnccn2)=O)C1 C1(C)(CNC(CC(=C)C)=O)CCN(C(=O)Cc2ccc(Br)c(Cl)c2)CC1 c1(C(N(CCCCN(C(COCC(C)C)=O)C)C)=O)cccc(F)c1C1CC1 c1(OC)cc(C(=O)NC2CCCC2(C)NC(c2cc(OC)n(C)n2)=O)nn1C n1(C(C)(C)C)nnc(CNC(C2CC(CNc3ccccc3)C2)=O)n1 C1(N(C(CCCCCC)=O)CCC)CC(NCCOC(C)(C)C)C12CCCC2 C12(CCNC(c3cc4n(c3)CCC4)=O)CCC1CN(C(=O)CC1(C3CC3)CC1)C2 CC1CCCCC1(CNC(=O)COc1cccc(Cl)c1)NC(=O)CCCF C(c1cccc(Cl)c1)=CC(=O)NCCC(c1ccccc1)OC C(=O)(C(C)(O)c1ccccn1)NCCC(C)NC(c1ccc(Br)o1)=O c1(C(=O)NCC2COCCN2C(C2CC(CF)C2)=O)cccc2[nH]ncc12 C1(S(C)(=O)=O)(C(=O)NC(C(C)NC(c2c(C)nc[nH]2)=O)CO)CC1 c1(NC(=O)C(C)OCC(F)(F)F)c(F)cc(Cl)cc1F.C12CCC(CC1)N2CC C1(C)(COC(C2CCN(C(CC(CC)CCO)=O)CC2)=O)CCC(=O)N1C N1(C(C(CC)OC)=O)CCC(C2(NC(=O)CC3CC(C)(C)OC3=O)CCC2)CC1 c1(C[N+](C2(CO)CCC2)([O-])OCCOCC)cc(Cl)ccc1Cl CC1(C)COCCC1C(=O)NCC1CC2CCC1N2C(=O)C(C1CCOCC1)O C(=O)(C(CO)C(C)(C)C)N1CCCCC(CNC(CC2CCC(C)(C)CC2)=O)C1 C1(COC)(CO)COCCN1C=O.n1(CC)cc(CCC(c2ccccc2)=O)nn1 C(=O)(C#CC1CCOCC1)N1CCC(CCNC(CC(C)SC)=O)C1 C(=O)(C(F)(F)C(O)CC)N(CC(CC)NC(c1cnn(CCO)c1C)=O)C N1(CC)C2CCC1CN(C(=O)CC13CCC1CN(C(=O)C(C)(C)CN(C)C)C3)C2 CCCC(CC(=O)Nc1ccc(CCF)cc1)NC(=O)C(F)(F)COCC c1(C(N2CCC(NC(CN(C)CC)=O)(CF)C2)=O)ccc(O)cc1[N+](=O)[O-] C(C)(C)(CCCC(=O)NCC(=O)NCc1nc(C#N)cs1)OC N1(C(c2c(CC)onc2)=O)CCC(CN(C(c2sccc2F)=O)CC)CC1 N1(C(C(CCOC)C)=O)CCC(C)(NC(c2ccsc2C)=O)CC1 C1(C(=O)NCC(C)(CO)NC(=O)C=Cc2cc[nH]c2)CCn2nnnc2C1 C=CCC(CNC(C1CCCC(=O)N1)=O)C(=O)NCC(C)(F)F N1(C(C2CC=C(C)CC2)=O)CCC2(CC1)CC2C(N1CC(F)(F)C1)=O c1(CC(N2CC(NC(C3CCC(CC)O3)=O)C2)=O)ccc(N2CCCC2=O)cc1 n1(C(C(N2C(CNC(CN(C3CC3)CC)=O)C=CC2)=O)C)cnc2ccccc12 N1(C(c2onc(CC)c2C)=O)CCN(C(c2cc(N)ccc2Cl)=O)C2(CC2)C1 C1(CNC(c2ccc(Cl)s2)=O)CC2(CN1C(=O)CC1CC=CCC1)CC2(F)F C1(C(N2CCC(C)(CNC(c3ccnn3C(F)F)=O)C2)=O)CCC2(CCC2)O1 Cc1ccc(Cl)c(C(=O)NC2CC2NC(c2cn(C)ccc2=O)=O)c1 CCCCS(=O)(=O)CC(=O)NC1CCC(CNC(C2CC23CC3)=O)C1 C(=O)(C(C)(C)C(C)(F)F)NCC1CN(C(C(COCC=C)c2ccccc2)=O)C1 c1(C(C(=O)N(C)CC2CCN(C(C3(C(F)(F)F)CC3)=O)C2)(F)F)ccc(F)nc1 C1(C(=O)N(C(CNC(c2ccc(C)o2)=O)C2CC2)C)(COC)CC=CCC1 N1(C(c2cc(C(C)C)nn2C)=O)CC2C(C1C(N1CCNC(=O)CC1)=O)C2(C)C c1(C(C)NC(C(=O)NCC)=O)ccc2c(c1)CN(C(=O)Cc1ccc(Cl)s1)C2 N1(C(C2CC(C)C2)=O)CCC(C)N(C(c2n[nH]c3ccccc23)=O)CC1 c1(C(=O)NCC2CN(C(CCC3C(C)(C)C3)=O)CC2O)ccc2c[nH]nc2c1 CCC(C)CC(C)CC(C)C(=O)NNC(=O)Cn1cc(Cc2cccc(C#N)c2)nn1 CC1CN2CCN1CC2CNC(=O)Nc1cc(N2CCOCC2)nc(Cl)c1 c1(C(=O)NC2CN(C(C34OCC(CC)(C3)C4)=O)CC2C)c(Cl)ccc(F)c1N C1(C(=O)NC(C(=O)OC)Cc2csc(Cl)c2)C2Cc3cc(Br)ccc3C12 C(c1ccc(C)nc1)=CC(=O)N(C1(CC=C)CCN(C(=O)C(CC)CC)C1)CC Cc1nc2ccccn2c1C(N1CC2C(C1)N2C(c1cc(Br)cnc1Br)=O)=O c1(CCNC(C(COC)n2cc(C3(C)CC3)nn2)=O)cnccc1F C(=O)(C(O)C(C)(C)CC)NCc1cn(CC(=O)NC2C(C=C)COC2)nn1 Cc1ccc2c(N(CC(=O)N(C)C)C)nc(N(C)Cc3cccnc3)nc2c1 C1(C2(O)CCC2)(CC2CCN(C3CCN(C(=O)OC(C)(C)C)C3)C2)CC1 CCC(C)(COC)C(=O)NC(C)C(=O)N(C12CC(C1)C2)C C1(NC(C(C)NC(C)(C)C)=O)CN(C(C2(F)CCC(F)(F)CC2)=O)CC1(C)C c1(OC)ccc(Br)c2[nH]c(C(=O)NC(C)(C)C#N)cc12 Cc1cc(N(C)C)ccc1C(=O)NC(C)(C)C(C)NC(=O)CN(C)S(N)(=O)=O N1(C(C(C(C)C)F)=O)CCN(C)C(CNC(c2ccns2)=O)C1 N1(C(Cn2ncc(CC)c2)=O)CCc2sc(-c3ccn(C)n3)nc2C1 C1(NC(C(C(C)C)C(C)C)=O)CN(C(c2ccnn2C)=O)CC2(CCOCC2)C1 N1(C(c2c(CC)nn(C)c2)=O)CC2CCCN(C(=O)C#CC3CC3)C2C1 C1(NC(c2cc(C)sn2)=O)CCSC12CN(C(=O)CCCC(F)(F)F)C2 C1(CNC(C(c2cccc(Cl)c2)N(C)C)=O)CCCCN1C(c1cnc(Cl)[nH]1)=O C1(C(=O)NC(C(=O)OCCC)C)CSCN1C(=O)Cc1ccoc1C S(=O)(=O)(c1ccccc1F)N1CCC(NC(Cc2c(OC)cc(Cl)cc2)=O)CC1 C=CC(C)(CC)C(=O)NC1CCCCN(C(C2(OC)CCC2)=O)C1 C1(NC(C2CC(C)C2(C)C)=O)CCC2(CC1)CC(NC(c1ncc(F)cn1)=O)C2 N1(C(C2CC(C)C2)=O)C(C(=O)NCCc2ccnn2C)CCC12CC2 CC(CC(F)(F)F)NC(=O)C(F)C1CC(NC(C2(C=C)CCCC2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1CCC(NC(CSc2nnc(C)o2)=O)C1 CCC(C)CC(C)C(=O)NC(c1cn(C)nn1)C(=O)NCC(F)(F)C(C)(C)O C1(NC(c2coc(Cl)c2)=O)CCN(C(C2CC(F)(F)C2)=O)CCC1(F)F N1(C(C2CC(C)=C(C)CC2)=O)CCC2C(C1)CN2C(c1ccc(O)nc1)=O O=C1CCc2cc(C(=O)NCC3(O)CN(Cc4cc(Cl)ccc4Cl)C3)ccc2N1 C1(C(=O)NCCCN(C(c2ccc(Cl)c(F)c2)=O)C2CC2)CC2C(C1)C2(F)F c1(CC(N2CC(C(N3CC(CC(C#C)C)C3)=O)C(C)C2)=O)ccccc1C#C N1(C(c2c(OCC)cccn2)=O)CCC(C2CN(C(=O)CC3CC3(C)C)C2)CC1 C1(NC(C(C2CCCC2)OCC)=O)CC(C)(NC(=O)Cc2ccc(Cl)s2)C1 C(=O)(C(F)(F)CO)N(CC(CC)NC(c1n[nH]cc1F)=O)C N1(C(C2(OCC)CCC2)=O)CC2CCCC(NC(=O)C(C3CCOCC3)C)C2C1 C12(CO)COCC1CN(N1CCCC(C(C)CO)CC1)C2.C(=O)CCn1cccc1 Cc1cc(=N)[nH]cc1C(N1CC2C(NC(c3cnc(C(C)C)nc3C)=O)C2C1)=O c1(OC(C)C)ccc(C(N2CCCC(CCNC(=O)C(C)(F)F)CC2)=O)c(Cl)c1 C1(CNC(Cn2nnc(C)n2)=O)CN(C(=O)CN2CCCS2(=O)=O)C2(CCC2)C1 Cc1cc(-n2nc(Cc3ccccc3F)nc2C2C(C)C2(F)F)cc(Br)c1 C1(CC(=O)N(C)CCN(C)C(c2ncoc2C2CC2)=O)CC(=O)NC(=O)C1 C1(CNC(C2C3COCC23)=O)CC2COCC2N1C(c1cccnn1)=O c1(C(=O)NCC2CC(C)N(C(c3cnco3)=O)C2)cnc2ccccn12 c1(C(=O)NCC(C(=O)NC2(CC=C)CCCC2)CC2CC2)cccc(O)c1C N1(C(C(C)C#N)=O)CC2(CC2)CC1CC(=O)NC1CC(C2CCC2)C1 CN1CC(O)(CN(C)C(C2CC2C(C)NC(C2(F)CC=CC2)=O)=O)C1 C(=O)(C(CC(C)C)NC(C1CCC2CC12)=O)NCC(C(CC)C)C C12(C(=O)OCC)COC(CNC(=O)C(CC3CCCC3)OCCNC(C)=O)(C1)C2 C1(NC(C2CCN(c3c(C)cccc3)CC2)=O)CC2(CNCC(=O)N2)C1 CCC(CC)C(=O)NC1(C)CC(NC(c2coc(-c3ccsc3)c2)=O)C1 C(=O)(C(C)C(C)CC)NC1(c2nn[nH]n2)CCN(C2CCCC2CC)CC1.C=CC Cn1c(C#N)cc2c1CCN(S(=O)(=O)c1ccc(OCC(F)(F)F)cc1)C2 N1(C(C=C2C(C)(C)CCCC2)=O)CCCC12CCN(C(=O)C=CC(F)(F)F)C2 C(=O)(CC(C)(F)F)N(CCCNC(C1(NC(C)=O)CCCC1)=O)CC N1(C(C2(CC#C)CCCCO2)=O)CC2(C1)CN(C(=O)Cc1ccnn1C)C2 c12cc(ccc1F)C1CC1C(=O)N2.c1(SC)ncc(C(F)(F)F)[nH]1 N1(C(c2c(C)[nH]nc2Br)=O)CCCN(C(=O)CCC2CCCN2C)CCC1 CON=CC(=O)NCC1CCCN1C(c1csnc1OC)=O CCC(C)C(O)C(C)C(=O)NCCCCN(C)C(C1CC1C)=O Cc1cccc(F)c1C(=O)NC(C)(C)CCC(=O)NC1(n2cncn2)CC1 C1(C(COC)C)CCN(C(=O)NC2CC(F)C(=O)N2)CC1 CC1C(CCc2ccccc2)NCC(C)(C)N1.c1(C(=O)OC(C)(C)C)cn[nH]c1 C(c1nc2ccccc2[nH]1)=CC(=O)NC(CNC(C=CCCC(C)C)=O)C1CC1 C(C(C)(C)CC(=O)N1CCOC(CN=[N+]=[N-])C1)NC(c1cc(C)ncn1)=O C1(N(C(C)(C)C)CCNC(C(C)Cc2ccncc2)=O)CCCC1C#N C1(NC(c2c(C)n(C(C)C)cc2)=O)CN(C(=O)CS(C)(=O)=O)CC12CC2 CCCCC(C)(C)NC(=O)CC1CCN(C)C1=O.C12CCCC1CNC2=O C(=O)(C(F)(F)CC1CC1)N1CC(CC=C)(NC(C2CC2C(C)C)=O)C1 CC1CCC=C1C(=O)N1CCN(C(=O)CCF)CC1C(F)F C#CC1CCCCN1C(=O)CCC(C)(C)NC(c1ccsc1OC)=O c1(NC(C2N(Cc3nc(CC(=O)OC)on3)CCC2)=O)cccnc1Br c1(C(N2C(CC(=O)NC(CC=C)(C)C)COCC2)=O)c[nH]c(C)cc1=O C(=O)(C1=NOC2COCC12)N1CCCC(C)(C(=O)NCCc2n(C)ncc2)C1 C(=O)(C(CC(C)C)C(C)C)NCCN(C(=O)CCNc1ccccc1Cl)CCC C1(CNC(C2(CNC(c3ccc(OC)cc3)=O)CC(=C)C2)=O)C2CCCCC12 Cc1cc(C(=O)NCC(C)(O)CNC(C2CS(=O)(=O)C2)=O)cc(C)c1O c1(CCCC)cc(C(N2CC(CC(C)NC(=O)C(CC)OC(C)=O)C2)=O)c(C)o1 CCCC(C(O)C(=O)NCC(C)(C)O)NC(=O)C=CC(=O)NC1CC1 c1(CC)sc(C(=O)NCc2ccc(CNC(=O)C(C)(C)SC)cc2)cc1C c1(C(=O)NC(CC(C)C)CNC(c2cc(C#N)c[nH]2)=O)cccc2c1OC(C)C2 Cc1ccc(F)c(C(=O)NC2CCCN(C(=O)CC3CCCSC3)CC2)c1Cl c1(C(=O)NC(C)C(CO)NC(=O)C2=CCCS2)ccc2nc(N(C)C)[nH]c2c1 C1(C(N(CC(CC)NC(=O)COCCOCCOC)C)=O)CC2(C1)CC2F c1(NC(c2cc(C)c(=O)n(C)c2)=O)nc(C(=O)N(C)C)n2ccccc12 c1(NCCCCC(C)NC(CCn2c(C)csc2=O)=O)ncc(Cl)cc1[N+](=O)[O-] C(=O)(CC(C)(C)O)N(CCCNC(C1(CC)COC1)=O)CCO C1(C(=O)O)CCc2nc(NCc3cn(C4CC5OC4C4CC54)nn3)nn2C1 CCC(C)C(O)C(=O)NCC1CN(C(c2sc(COC)nc2C)=O)CC1O Cc1ccc(OCc2occ(C(=O)NC(C)C(n3cc(CO)nn3)C)n2)cc1 Cc1cccc(Br)c1CC(=O)N(C1CC1)CC1CC(O)C12CCC2 N1(C(CCC#CC)=O)CC23CCCC2(C1)CN(C(=O)CN(C)C(C)=O)C3 N1(C(c2cnc(CC)[nH]2)=O)CCC(CNC(=O)Cc2ccc(F)cc2F)C12CC2 C1(C(N(C2CCN(C(=O)C=Cc3nnn(C)n3)C2)C)=O)CCCCN1C CC1CCC(NC(C2(C)CCC2)=O)CN1C(=O)CO C1(C(N(C(C)CNC(=O)C(C)C2CCC2)C)=O)CCCC(C(F)(F)F)C1 Cc1nnc(SCCCc2cccc(Br)c2)c(NC(=O)CCC2CCC(C)C2)c1C C1(C(F)(F)F)(C(=O)NCC(C)(C)OCCNC(C(=O)N(C)C)=O)CC=CCO1 N1(C(c2ccc(C3CC3)s2)=O)CCN(C(=O)CC2CCCC(O)C2)C2(CCC2)C1 c1(C(=O)OC)ccc(C(=O)NCCCCNC(=O)C(c2ccccc2)OC)nc1 C1(NC(c2cnc(COC)s2)=O)CC2CCC1N2C(=O)C1=NOC(C(C)(C)C)C1 C12(NC(=O)C3=CCC3)CCN(C(C34CCN(CC3)CC4)=O)CC1C2 c1(C(=O)NC(CC(C)NC(c2cc(C(C)=O)c(C)o2)=O)C)cn2c(n1)CCC2 N1(C(C(C2CCC2)OC)=O)CCN(C)C(c2cn(CC(F)(F)C(F)(F)F)nn2)C1 N1(C(c2c(CC)n(C)nn2)=O)CCC(C)C(NC(=O)Cc2nnc(S)s2)C1 c1(C(N2CCCC(CN(c3nccc(C#N)n3)C)C2)=O)ccc2ccn(C)c2c1 C1(CC(N2CCCC(NC(c3c(SCC)nccn3)=O)C2)=O)CCCCC1(F)F c1(OC)ccc(Cl)nc1C(=O)N(CCNC(C1C2C3CCC(C3)C12)=O)C1CC1 C(CCCCC(=O)N(C1CCN(C)C1)C)C(CN(C)C)C(=O)NC1CC1 N1(C(CCc2c(C)ncs2)=O)CC(CNC(c2csc(CO)n2)=O)CC1(C)C C(C(C(=O)NCCCCCC(C)C)C(C)C)NC(c1c(C)c[nH]n1)=O c1(C(N(C2CC(NC(=O)C=CSc3ccccc3)C2)C)=O)ccsc1S(N)(=O)=O c1(C(N(C)CC2(NC(c3c(OC)csc3)=O)CC2)=O)cc2ccccn2c1 C1(NC(CC(CC)C2CCC2)=O)CC=C(C(=O)NCCC2CCOC2)C1 c1(OC)ccc2c(n1)NC(C(N1CCC(C(C)NC(=O)CCCCCl)CC1)=O)C2 c1(C(=O)NCCC(C)(C)NC(c2ccc(OCC)cc2)=O)cc2sc(C)nc2[nH]1 C1(CNC(CCCOC(C)C)=O)CC(NC(c2cc3sccc3s2)=O)C12CCC2 N1(CCCC)CCOCC1C(=O)N(CCCCCCNC(=O)C(CC)OC)C c1(C(=O)NCCN(C(C=Cc2ccc(CC)o2)=O)C(C)C)ccc2nnnn2c1 c1(OCC(N2CCC(F)(CNC(=O)COCCF)C2)=O)ccc(F)c(C2CC2)c1 C1(NC(CC2(COC)CC2)=O)CN(C(C2C(F)(F)C23CCC3)=O)CCC1CO C1(NC(CC(C)C2CC2)=O)CCC2(CC1)CN(C(c1cccc3ncnn13)=O)C2 c1(OC)ccc2cc(C(=O)NCC(C)N(C)C(c3cc(CF)on3)=O)ncc2c1 c1(C(N2C(C(=O)NCCCN(S(CC)(=O)=O)C)CCC2)=O)cncc(N)n1 Cc1nc(CCC(=O)NC2C=CC(CNC(=O)C(F)n3ccnc3)C2)cs1 Cc1nc(C(=O)NCC2CC(NC(c3ccnc(C(F)(F)F)n3)=O)C2)c(C)n1C c1(C(N(C(c2cn(CCCN3CCCC3)nn2)(C)C)C2CC2)=O)nc(Cl)c(Cl)s1 Cc1c(C(N2CCC(NC(=O)C(F)n3cccn3)C2C)=O)[nH]c2c(Cl)cccc12 c1(C(N2CCC(OCCO)C2)C(=O)Nc2ccc(C)s2)cc2ccccc2o1 N1(C(C(COC)O)=O)CCC(CO)(CNC(=O)C=Cc2ccc(C)o2)C1 c1(CNCC2N(C(=O)Cc3sc(O)nc3O)CCC2)ncc2c(n1)CCOC2 C1(C(N2C(C)(CC)CC2)=O)CN(C(=O)CCCC2CC2)CC(F)(F)C1 C1(NC(C2OCC(C)C2)=O)CC1C1CCCN(C(C2(C#N)CC=CC2)=O)C1 c1(CN2CCC(C(C)NS(CCCC)(=O)=O)C2)cc(F)ccc1OC N1(CC(=O)NC2CC(CNC(C(C)=CC)=O)C2)CC2CC2C1 CCC1=NOC(C(=O)NCC2COCCN2C(c2nc(C(F)(F)F)sc2C)=O)C1 CCCC(C(=O)N1CC(NCC)C(C)C1)NC(C)=O CC1(C(N2CC(CNC(C3(n4nccn4)CC3)=O)C2)=O)C2Cc3ccccc3C12 Cc1cc(C(=O)NCCNC(=O)C(=O)NC(CO)C(=O)O)ccc1O.C(=O)N c1(OC)c(C(=O)NCc2cccc3cccnc23)cccc1[N+](=O)[O-] Cc1cnc(C)c(C(=O)NCC(C)(O)CNC(C2CC(F)(CO)C2)=O)c1 N1(C(c2ccc(CCC)cc2)=O)CCC(C)C(NC(=O)Cn2cccc2)C1 C1(NC(CCC(=O)N(C)C)=O)CC12CCC(NC(C1CCCC1(F)F)=O)CC2 CCCCCCC(=O)NC1CCCN(Cc2ccc(F)cc2)CC1 C(=O)(CP1(=O)CCCCC1)N1CCCC(CCNC(c2c(C)cnnc2)=O)C1 CCC(CC)C(C(=O)N1CCC(CN(C)C(C2CCCCC2)=O)C1)OC c1(OC)cc(OC)c(Cl)c(C(=O)N(C(C)CN(C(=O)CCCCC(C)C)C)C)c1 C1(C(=O)NC2CN(C(CC(c3c(C)n[nH]c3C)C)=O)CC2O)CC(=O)NC(=O)N1 C1(=CCNC(c2scc(C(C)(F)F)n2)=O)CCN(C(=O)Cc2cncnc2)CC1 Cc1cn(C)nc1CNC(=O)CC1(CNC(=O)CN2C(C)CCC2C)CC1 C1(CC(=O)NC(C(=O)OCC)C)CN(C(=O)C(C(C)O)N(C)C)CCO1 C(C(C(=O)NC(C)(C)C)n1cc(-c2ccncc2)nn1)O.C1(C)CCN(CC)C1 Cc1c(C2CC2NC(=O)CC#N)cccc1Br.C12(CCCC1)C(=O)NC2 Cc1ccsc1C=CC(=O)NC1CC(NC(=O)C(c2ccccc2)C2CC2)C1 c12ccc3c(c1)CCN(C3)C2=O.N12CC3(CCC3)C1C2=O.CO.OC CN1C(=O)CCC1CC(N1CCN(CC(=O)NCC2(c3cc[nH]n3)CC2)CC1)=O N1(C(C=CC(C)C)=O)CCC(CNC(C2CC2C(C)(F)F)=O)C(O)C1 c1(OC(C2CCCC(NCC3CC(OC)CN3C)C2)=O)ccc2cccnc2n1 CC1CN(C(c2cccc(C(N)=O)c2)=O)CCC1CNC(=O)Cn1nnc(=N)[nH]1 c1(-c2nc(N3CCC(N(C(CCCCCC)=O)C)C3)sn2)ccccc1[N+](=O)[O-] C1(F)(C(N2CCC(OCC)C2)=O)CCN(c2cc(OC)ncn2)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCCCCCN(C(C=C(CC)CC)=O)C N1(C(c2cn(CC)nn2)=O)CCCC2(CCN(C(C3CC4CC4CC3C)=O)C2)C1 C1(NC(=O)CC2CCCC2)CCC12CCN(C(C1CS(=O)(=O)C1)=O)CC2 C(=O)(CC(C)CC(C)(C)C)N(C)CCOCCNC(c1ccc(Br)c(N)n1)=O c1(C(=O)NC2CN(C(c3cc(OCC)n[nH]3)=O)CC2O)cc(C)ccc1F c1(C(=O)NCC2CN(C(C3CCCCO3)=O)CCO2)ccc(O)c(F)c1 Cc1c(F)ccc(C(N2CC3CC3(NC(=O)C(C)CC3CC3)C2)=O)c1C C=CCN=C(NCc1ccco1)NCc1cn(C(C)(C)C)nn1 C#Cc1cccc(C(=O)N(CC(CC)SC)CCNC(=O)C=CCO)c1F CCC(CC(=O)N1CCCC1C1(NC(C2CN(C(C)=O)C2)=O)CC1)CC(F)(F)F c1(C(N2CCC(CN(C)C)C2)C(=O)NC2CCCCC2)cc(F)c(Br)cc1F c1(C(=O)NCC=CCNC(CC2COCC(C)O2)=O)cc2ccsc2n1C C1(C)(COC)CC(NC(=O)CNC(C)=O)CN1C(c1cc2n(c1)CCC2)=O c1(OCC)ccc(CC(=O)N(C2CCN(C(C3(C)CCCOC3)=O)CC2)C)cc1 c1(OC)cc(C(=O)NCC2(C(=O)Nc3scnc3C(N)=O)CC2)c(Cl)cn1 N1(CC)OCC(=O)N(C(=O)OC(C)(C)C)c2cccc(Br)c21 Cc1ccnn1CC(=O)NC(C)C(C)C(=O)NC(C)(C)C(O)CO C(=O)(CCCCCCN=[N+]=[N-])N1CCCC(F)(CNC(C(CC)O)=O)C1 N1(C(C2C(C=C)OCC2)=O)CC=C(CNC(=O)C(C)(F)F)CC1 c1(CC)[nH]nc(C(=O)N(C2CCN(C(=O)Cc3ccc(C)nc3)C2)C)c1[N+](=O)[O-] c1(C(N2CC(CCCC)N(C(=O)C(C)CSC)CC2)=O)cc2ccccc2o1 CC(CCNC(=O)CC(O)c1ccccc1)CCNC(c1coc(C2CC2)n1)=O C(=O)(C1=CSCS1)NCC(C1(O)CN(C(C2CC2c2ccc(F)cc2)=O)C1)(C)C n1(CC)ccc(C(N2CC(C)(NC(=O)CC3CCC(C)C3)C2)=O)n1 C1(C(N2CCN(C(c3cccc(C)c3N)=O)CC2CF)=O)CC2CCC(C1)C2O C1(COCC(=O)NC2(c3ccncc3)CC2)(COC)CCN(C(=O)CC2CC2)C1 C(=O)(C1CCCn2nccc21)N1CCCN(CCNC(C(=O)NC(C)C)=O)CC1 CC(CC(=O)N(C1CCC(CNC(=O)C(C2CCCCC2)O)CC1)C)C(C)(C)C c1(CC(N2CC(CCNC(=O)C(O)CF)OCCC2)=O)c[nH]c2ncccc12 C1(C(C(=O)N2CC(N(C(=O)C=CCCOC)CCO)C2)OC)CC(F)(F)C1 C1(C(=O)Nc2cc(OC)c(F)cn2)CCCC12CCN(Cc1ccnc(C)c1)C2 N1(C(C(F)OC)=O)CC2(CCN(C(=O)CN3CCN(C)CC3)CC2)CC1C CC1(C)OC2CC(C(=O)NC3(CO)CCN(C(C4COCCO4)=O)C3)CC2O1 c1(C(N2CCC(C)(CNC(C3(Cl)CC34CCC4)=O)C2)=O)cc(N)c(F)cc1F C#CCCCCC(=O)N1CC2CC(C(NCP(C)(C)=O)=O)(C2)C1 C(=O)(CCS(C)(=O)=O)N(C)CC1(NC(C2CC(=C(F)F)C2)=O)CC1 c1(C(N(CC(O)CNC(c2cnc(N(C)C)nc2)=O)C)=O)cc2cccnn2c1 C1(NC(C2N(C(N)=O)CSC2)=O)CC2CC(C1)N(C(=O)C(F)(F)C1CC1)C2 C12(C(N(CC=C)CCOC)=O)CC(CN(C(=O)CCCC(=O)C3CC3)C1)C2 C1(C(=O)NC2CC(C(N(CC(COC)(C)C)C)=O)C2)C2CCC(F)(F)C12 Cc1c(C(N2CCCC2CNC(c2cn(C)nc2C2CCCO2)=O)=O)ccn1C c1(C(C(=O)NCc2ccco2)N(C(CC)C(=O)OC)C)cc(OC)ccc1Br N1(C(C2CCCC(OC)C2)=O)CCCC(NC(=O)Cc2cnn(C)c2)C1C c1(C(=O)NCCCNC(c2n(CC=C)ccc2)=O)cc(N(C)C)ccn1 c1(NCC2CC(=C)C2)nc(=NC2CCCC(SC)C2)[nH]c2c(C)nn(C)c12 N1(C(C2(F)CCN(C(c3cccc(F)c3)=O)C2)=O)CCn2ccnc2C1 N1(C(C=COCC)=O)CCN(CCOC2CCN(C(=O)C(C)C)C2)CC1 C(N=c1cc(C2CC2)nc[nH]1)C12N(C(c3cc(CCC)on3)=O)C(CC1)CC2 CC1(C)CC2(CC(C(=O)NCC3C4CN(C(C5CC=CC5)=O)CC34)C2)C1 c1(-c2cc(C)c(C#N)cc2)ccc2ncc(C(=O)NCC3(C)OCCO3)n2c1 N1(C(c2cc(C)sc2C)=O)CCCC(CC(N2CCC(C3CC3)C2)=O)CC1 C1(NC(C(C)OC)=O)CC12CCN(C(c1ccnc(F)c1Cl)=O)CC2 N#Cc1cc(C(=O)NCCOCCNC(C2(F)CCSCC2)=O)co1 c1(SCC(=O)NCC(CO)NC(c2ccnn2CCF)=O)nnc(S)s1 Cc1cccc(C(F)(F)C(=O)NC(C2CCCN(CC3(C4CCC4)CC3)C2)=O)c1 C(=O)(C1=CCCSC1)N(CCNC(c1cnc(C(C)(C)C)s1)=O)CC1CC1 N1(C(CNC(c2c(C)onc2)=O)=O)CC2(NC(=O)CN3CSCCSC3)CC1C2 C1(OCC)CCCC1C(=O)NC(C(=O)NC1CC(CCF)C1)C1CCCO1 N1(C(COC)=O)CCCC(NC(c2c(C)nsc2Br)=O)C1C CC1CCCC1C(=O)NCC1(O)CC(CNC(=O)CC2CCCC2)C1 C1(C(N(CC(C)CNC(c2cscc2Br)=O)C)=O)Cc2nncn2C1 c1(C(=O)OCC(c2ccc(C(=O)OC(C)(C)C)cc2)=O)cnc2n1CCCC2 C1(C(=O)NCCC2(O)CCN(C(c3ccc[nH]3)=O)C2)Cc2nccn2C1 c1(OCCOC)ccc(C(=O)NCC#CCNC(=O)CCc2ncc(C)[nH]2)cc1 CCCC(C#N)C(=O)NCC1(C(=O)N(C(C)CO)C)CC1 O=C(C1CCCc2scnc21)NC1(CCNC(c2cscn2)=O)CCC1 C1(NC(C(CNC(C(CC)n2ccnc2)=O)(C)C)=O)CCN(OC)CC1 C1(CCCNC(C(CC)NC(C)=O)=O)CCCCN1C(C1CCS(=O)CC1)=O c1(C2CC(NC(C(C)NC)=O)C2)ccc(Cl)c(Cl)c1 C1(OC)CCC(NC(C2(C(C)NC(=O)CC3(C)CCOC3)CC2)=O)CC1 C(C(CC(F)(F)F)NC(=O)CCCNC(c1cccnc1)=O)NC(C1C(C)C1C)=O C1(C(=O)NCC(N2CC(CC)NCC2)=O)CCOC(=O)CC1 C1(N(C(=O)C(C2CCOCC2)O)CCOC)CCN(C(c2ccoc2)=O)CC1 C(C(F)C(=O)NC1CC1CNC(C1(O)COC1)=O)NC(=O)OC(C)(C)C c1(C(=O)NCC=CCNC(C2CCC(C#N)CC2)=O)cccc2ncsc12 C(CC(C(=O)Nc1cn(C)nc1OC)NC(=O)CC1CC2CC2C1)=CC C1(C(N(CCNC(=O)C(C)(C)c2ccns2)CC)=O)C(F)(F)C12CCC2 C(C(F)(F)C(C)(C)O)NC(C1N(C(c2c(OC)cncc2)=O)CSC1)=O c1(C(=O)NC2C(CNC(Cc3c(C)con3)=O)CCC2)cccnc1C1CC1 C1(N(C(C2CC(SC)C2)=O)C)CCN(C(c2ccc(O)nc2)=O)CC12CC2 N1(C(=O)NCC2(SC)CCCC2)CCC2(O)CCCCC2(O)C1 C(=O)(C(C)NC(=O)C(C)N(C)C(C)=O)NCCOC CCC(CN=c1cc(NC(c2ncc[nH]2)C)nc(C)[nH]1)OC Cc1cc(C(N2CCCC2C=CC(=O)NCCC(O)C(C)C)=O)c(C)n1C n1(CC)cnc2[nH]c(=NC(C)CCC3CC3)[nH]c(=NC(C)c3cc(COC)no3)c12 N1(C(=O)CN2C(=O)CNC2=O)CCC2CN(C(c3ccc(O)cc3F)=O)C2C1 C=CCN(OC)C(=O)C1=NOC(CNC(=O)CCNC(N)=O)C1 C(=O)(C1CCCc2ncnn21)N1CCCC(NC(C(C(C)O)N(C)C)=O)CCC1 C(CCCC(=O)O)NC(=O)NCC(C)C.c1(C(=O)OC)cn(Cc2ccccc2)nn1 c1(C(=O)NC2CC(n3cc(CCC)nn3)C2)c(CSc2ccccc2)noc1C CC(=O)CC(C)(C)C(=O)N(CCCn1cc(-c2cc(F)ccc2Cl)nn1)C N(C1COc2cccc(F)c21)C(=O)NC1C(C)(CC)C1 C12(C(=O)NCC3(CNC(c4ccc(C)s4)=O)CC3)CC(CC(C)O1)C2 C1(CNC(C2(C)CN(C(C)=O)C2)=O)CCCCN1C(=O)C(C)CC1CCC1 C(=O)(C(C(C)(C)C)NC(N)=O)NCC1N(C(c2c(C)nsc2)=O)CCC1 C1(C(=O)NC(CNC(c2c(C)ccc(C)n2)=O)(C)C)CN2CCC1(C)CC2 CCC(C)C(O)C(C)C(=O)NCCCN(C(=O)C(C)CC1CCC1)C CC1CC(CC(=O)NCCc2ncc[nH]2)CN1C(=O)CC1CC1 C(=O)(CN=c1[nH]c2ccccc2s1)N1CCC(NC(C(C)O)=O)C2(C1)CCC2 c1(CNCC2CCN(C(c3cccc(CC)n3)=O)C2)ccc(C)c(OC)c1 C1(CNC(C2C=CC(NC(=O)CCCCCF)C2)=O)CC2(CCCCC2)C1 C1(CN(C(CCNC(=O)NC)=O)C)CCCCN1C(=O)C=Cc1ccncn1 c1(C(N2CC(SC)C(n3cc(C(C)O)nn3)C2)=O)nc(C2CCC2)ncc1Br Cc1c(F)ccc(Cl)c1C(N1CC2C(NC(c3cccc(N)c3)=O)C2C1)=O CC(=O)C(C)CC(C)C(=O)NCCC(=O)N1CCC1CC(C)C CN1CCN(C)C(C(=O)NC2CCOC(NC(c3cc(F)ccc3F)=O)C2)C1 C1(CNC(c2ccnc(C(F)F)c2)=O)C2CN(C(C34CC(C(=O)OC)(C3)C4)=O)CC12 C1(NC(c2ccc(C#C)cn2)=O)CN(C(C2CCCS2)=O)CC2(CC2)C1 N1(C(c2cnc(CCCC)s2)=O)CC2CCOC2(CNC(c2cc(Cl)no2)=O)C1 C(C)(C)(CCCC1OCCO1)NCC(C)C(=O)OC(C)(C)C C1(NC(C(c2c(OC)cccc2)=O)=O)CC(C)CN(C(c2cscn2)=O)C1 C(CCS(C)(=O)=O)(C(=O)N1CCC(C)CC1CNC(c1cocn1)=O)OC c1(C(=O)OC)cccc(NC(C2CCCN(C(c3cc[nH]c(=N)c3)=O)C2)=O)c1 C1(CNC(CCSCC)=O)CC(C)N(C(c2csc(COC)c2)=O)C1 C#Cc1nc(C(N2CCC(NC(=O)C(C)Oc3cccc(C)c3)C2)=O)cs1 c1(CN(C(CSC)=O)C)ccc(CNC(C2(C)CCOC2C)=O)cc1 C(C#Cc1cn(C2CCCC(C(=O)O)C2)nn1)NC(c1c(C)ccc(C)n1)=O Cc1cn2c(C(=O)NC3CC4(CCN(C(=O)Cc5csc(=N)[nH]5)C4)C3)cnc2s1 C1(NC(CC(=C)C)=O)CC12CCN(C(c1cc[nH]c1C1CCC1)=O)CC2 C(C(COC)C(=O)NC(C)CNC(c1cc(CS(C)(=O)=O)on1)=O)OC CC(CS(C)(=O)=O)C(=O)N1CCC2CN(C(=O)C3=CCCC3)C2C1 N1(C(C(N2CCOCC2)C)=O)CCC(C2CCN(C(=O)C3=CCCCO3)CC2)C1 c1(NC(CC2N(C(C3CCC(C(C)C)CC3)=O)CCOC2)=O)nc2c(s1)CCC2 c1(C(N(C)CC2CCN(C(c3ncn(C)n3)=O)C2)=O)cc(C(F)F)n(C)n1 N1(C(C)=O)CCCC(C2CCN(CCN(CC(F)(F)F)C)C2)C1 CCC(C)CC(C(=O)Nc1cncc(OC)c1)NC(=O)C1=CCCCO1 C1(O)(CNC(C(=Cc2ccccn2)C)=O)CCCN(C(=O)C(O)C2CC2)C1 C1(C(=O)NC(C)COCCF)(CC)CCCN(C(C2CN3CCC2CC3)=O)C1 C1(CCOC)CN(C(c2ccnnc2)=O)CCN1C(c1ccccn1)=O CN(C)N=c1nc2scnc2c(N2CCC(n3cc(Cl)cn3)C2)[nH]1 CCC(CC)CCCC(=O)N1CCN(C(c2cccnc2OC)=O)CC1CC C1(CC)CCCCC1C(=O)NCC1(C(=O)NC2(C)CC=CC2)CCCO1 C1(NC(C23C(C)(C)C(CC2)CC3)=O)CCCC2CN(c3ncc(O)cn3)CC12 c1(-c2cn(CC3CC(C(N4CCCC4C4CC4)=O)C3)nn2)ccc(CCO)cc1 CC1CN(C(=O)C2=COCCO2)CCC1CNC(c1cnn2c1OCC2)=O Cn1ccc(C2(C(=O)NC(c3ccccc3)CNC(=O)CNC(N)=O)CC2)n1 C1(CC)CCC(C(=O)NC(C)CN(C(=O)CN(C2CC2)CC)C)CC1 N1(C(CC(C)C)=O)CCCC2CN(C(=O)C=C(Cl)Cl)CCC12 c1(CC(CN2CCSCC2)NC(=O)NCc2c(C)nns2)cccc(F)c1 C(=O)(C1=CCC(F)(F)CC1)NC1C(C)CCN(C(c2ccc(C)c(C)n2)=O)C1 C1(NC(c2cc3n(n2)CCO3)=O)C2CCN(C(=O)CCc3cc[nH]n3)CC12 C(=O)(C1=C(C)OCC1)N1C(CC(=O)NCc2ncc(CC)s2)CC(O)C1 N1(c2c(C)c(NCC(N3CCOCC3)C)ncn2)CCC2OCCC2C1 C1(C)(CC)CC(NC(c2ccc(Cl)o2)=O)CN1C(c1cc(C)c(Cl)cn1)=O C1(C(N(CC(=O)OCC)C)=O)C2CCC(C2)N1C(C1CC12CCOCC2)=O N1(C(C2(CCCC)CC2)=O)CC23CCCC2(C1)CN(C(=O)CCC(C)OC)C3 c1(NC(C2CCCO2)COC)nc(N2CCC(OC)C2)nc2ccsc12 C(N=C(NC1CC(OC(C)(C)C)C1)N1CCC(C)C(C)C1)NC(C)=O N1(C(COC)=O)CC(C)(C)C1C1CCN(C(c2sc(CC(C)C)nc2C)=O)CC1 C1(C(N2CCC(CCNC(C3(C(C)(C)C)CCC3)=O)C2)=O)CCc2nncn2C1 C1(NC(C2CC2c2cn[nH]c2)=O)CC2CCC1CN(C(C13CCCCC1C3)=O)C2 N1(C(C(c2ccc(F)cc2)CC)=O)CCC(NC(C2(CC)CC2)=O)C(CO)CC1 C1(NC(C(C(C)(C)C)O)=O)COC2C(NC(=O)C=CCN3CCCCC3)COC12 Cn1[nH]c(=N)cc1C(=O)NCc1nn(C)nc1Br N1(C(C2C(C=C)OCC2)=O)CC(C)OC2(CCN(C(=O)C3=CCCOC3)CC2)C1 Cc1cc(C(=O)NC2CCCC2CC(=O)NCC(C)(C)CO)no1 N1(C(c2c(COC)cccc2)=O)CCN(C(=O)C(O)CC(F)F)CC(C)(C)C1 c1(C=O)ccc(C(N)=O)c(Cl)c1.n1(CC(=O)NCCCN(CC)CC)cncn1 c1(OC)ccc(C)nc1C(N1CC(NC(c2cc(N)ccc2Cl)=O)CC1C)=O N1(C(c2cc(C)c(C(F)F)o2)=O)CC(C2CCCN(C(=O)C=C(Cl)Cl)C2)C1 C1(CC(=O)NC(CC)CSC)CN(C(c2cnc(SC)[nH]2)=O)CC12CC2 N1(C(C2CC(C)N2C(=O)C=Cc2cncn2C)=O)CC2C(C1)C2(C)C CCC(C)(C)C(C)CC(=O)NCC(C1CC1)NC(c1ccn(CCO)c(=O)c1)=O C(CC(=O)NC(C(N)=O)C1CC1)N(C(=O)CC1CCSC1)C c1(C(=O)NC2(C)CCN(C(C(CCSC)O)=O)C2)ccc2ccncc2c1 CC1CCC(Cl)=C(C(=O)N2CCN(C(C3CCC(=O)N3)=O)CC3(CC3)C2)C1 CC1CC(c2ccccc2)CCN1Cc1cn(-c2cccc(F)n2)nn1 C(=O)(CC(C)(O)CCC)NCCCC(CO)NC(C(C)OCCCC)=O CC1CC(C(=O)NCCCNC(=O)CCCNC(N)=O)CC(C)N1C(N)=O c1(C(=O)NCCC2CCN(C(C(CN(C)C)O)=O)C2)cc(F)c(F)cc1F N1(C(CCC(=C)Br)=O)CCN(C(=O)CCCC)C(c2ccnn2C)C1 Cc1ccc(CC(N2CCC(CCNC(=O)CCc3cscn3)CC2)=O)cc1O N1(C(=O)CN2CC3CC3C2)CCC2(CC1)CC(NC(C1(c3cc[nH]c3)CC1)=O)CO2 N(C(=NCCCCl)NCCSc1ccc(Br)cc1OC(F)F)C1C(=O)OCC1 c1(C(=O)OC)coc(C=CC(=O)NCC2CCN2C(c2c(CO)noc2C)=O)c1 c1(C(N2CCC(C)(NC(C(CCCC)O)=O)C2)=O)cc2cc([N+](=O)[O-])ccc2o1 CC1=C(C(=O)N2CCC(CNC(=O)C(C(C)C)c3cccc(Cl)c3)C2)CCO1 c1(NC(C2N(C(C(C)N(C(C)=O)C)=O)CCSC2)=O)cc(C(F)(F)F)ccc1Cl C1(CN(C(COCCN(C)C)=O)C)CCCN1C(c1cc(C(F)(F)F)no1)=O C1(C(N2CCCCC2CNC(C2(F)CCCOC2)=O)=O)(CC)CCC(O)CC1 C1(NC(c2cc(OCC)n[nH]2)=O)CCN(C(C2CCC2CF)=O)C12CCC2 Cc1nc(N(C2CNCC2F)C(c2cc(Br)ccc2C#N)=O)c2sccc2n1 C1(NC(CCOC)=O)CC2(CCC(CNC(=O)C(O)C(C(C)C)OC)CC2)C1 CC(C(C)(C)C(=O)NCC1(C)CC2CCC1C2)NC(C1CC2(CCC2)C1)=O c1(CCC(=O)Nc2[nH]c(C)c(C)c2C#N)ccc2c(c1)CCO2 c1(CC(=O)NC(CN(C(COCCOC)=O)C)C)cccc(N2CCCC2=O)c1 C1(=CCNC(CSC)=O)CCN(C(c2cc(-c3cccnc3)nn2C)=O)CC1 C1(CC(=O)NC2CCN(C(C3C(c4scc(C)c4)C3)=O)C2)CCCCCO1 C1(C(N(C(CC)C(N2CCN(CCF)CC2)=O)C)=O)CCC(=O)N(C)C1 C(=O)(C1CCCc2cnn(C)c21)N1CC(CC)C(NC(c2conc2C)=O)CC1 c1(C(C)C)ccsc1C(=O)N(C1CCCCC1)CCCC1CCC1 C1(Nc2ncnc(CC)c2F)CCC2(C1)CN(C(c1cccc(I)c1F)=O)C2 N1(C(CS(=O)(=O)NC)=O)CCC(CNC(C2C3CCCC23)=O)C(C)C1 C1(CN(C)C(C2CCCC23CC3)=O)CCCN(C(c2cccc(CC#N)c2)=O)C1 C1(C(=O)NC(C2CCN(C(C3CC3C)=O)CC2)C)CCC(NC(N)=O)CC1 C(N=c1[nH]c(N2CCN(CCC#N)CC2)nc2c1CCC2)C1(S(CC)(=O)=O)CC1 C(=O)(CCCSc1ccccc1)NCC(C)N(C(C1(C(C)(F)F)CC1)=O)CC c1(CNC(C2(C)CC2(Cl)Cl)=O)cnn2c1CN(C(=O)CC1CCCCC1O)CC2 CN1CC(C)(C)CC1C(=O)NCC1CCC1C(=O)NCC1(C2CCC2)CC1 S(=O)(=O)(c1cc(C(=O)O)cs1)N1C(C(=O)OC)CCOCC1 O=C(C1CCCc2sccc21)NC1CCOCN(C(=O)COc2cccnc2)C1 C1(C(=O)NCC#CCNC(c2c(C)[nH]cc2)=O)CCc2nnc(C)n2C1 Cc1c(N2CCCCC(NC(C3CC4(CCCC4)C3)=O)C2)ncnc1C(F)(F)F CC(CCC(C)(C)C)NC(=NCc1ccc(F)cc1)NCc1cnn(C2CC2)n1 CC1CN(C)CCC1NC(=O)C(Cn1cccn1)NC(c1cc(C#N)cs1)=O Nc1c(F)ccc(C(N2CC3CC2C3NC(=O)CCc2cccs2)=O)c1F c1(C(N(C2CCCN(C(=O)C3=CCSC3)C2)C)=O)ccc(C(F)F)c(F)c1 N#Cc1ccc2c(C(N3CCC(CNC(=O)CCC(F)F)C3)=O)c[nH]c2c1 N1(C(C(C)(C)F)=O)CCOC(CNC(c2cnc(C(=O)N(C)C)o2)=O)C1 c1(OC)cc(C)c(CN2CC3CN(C(c4ccc(Br)cc4C)=O)CC23)cn1 c1(OC)cc(F)c(Cl)cc1C(=O)N(C)CCNC(c1ccoc1)=O CCCC(C)(CC)C(=O)N1CCC2C(C(=O)NCc3ccncc3F)C2C1 CCCC(CC)CCC(=O)NC(c1c(C)cccc1Br)C(N1CC(C)CCCC1C)=O N1(C(C2(CC#C)CCOC2)=O)CCC=C(C(=O)NCC2CCCOCC2)C1 c1(C(=O)NC2C=CCN(C(CCSc3nc(C)[nH]n3)=O)C2)cc(C(F)F)ccn1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(NC(C=C(CCC)CCC)=O)C1 N1(C(C=CCOC)=O)CC(C(C(=O)NCC(F)Cl)OC)C1 O=C(C#CC1CCC1)NCC1CCCC(NC(C2(F)CC=CC2)=O)C1 S(=O)(=O)(c1cccnc1NC(c1ccoc1)C)NC(CC)CCN1CCCC1 C(CCCC(=O)NCC(C(C)C)NC(C1CC(c2ccccc2)O1)=O)SC c1(NCC2CC(=C)C2)cc(=NCC2CCC3CC2C3(C)C)[nH]c(C)n1 N1(C(c2cn(CCOC)nn2)=O)CC2CC(CNC(=O)CC3CCCO3)C(C2)C1 CC1C(C)S(=O)(=O)CCN1C(C1(n2cc(C3(O)COC3)nn2)CC1)=O c1(C(Cc2onc(-c3ccc(N)cc3)n2)=O)n[nH]c2cc(Cl)ccc12 C(Cc1ccccc1)(C(=O)NCC(C)(C)CN1CCCC1)OC N1(C(C2ON=C(C(C)C)C2)=O)CC2CCC1CN2C(C1COCCN1C(C)=O)=O CC1(C)CN(C(c2ccc(OC(F)F)cc2)=O)CCC1NC(=O)CCS(C)=O N1(C(CCCC(C)NC(c2cc[nH]c2C2CC2)=O)=O)CCc2ccc(F)cc21 N1(C(C(CNC(c2ccnc(O)c2)=O)CC2CC2)=O)CCCCC12CC2 c1(CN=c2[nH]c(C)c(C(N3CCCC(C)(O)C3)=O)s2)ccc(C2=CCCC2)cc1 C1(C(NOCC)=O)CCN(C(=O)C(CC(C)C)OC)CC1(C)C.Cc1nnc(CC)o1 c1(C(=O)NCC(CNC(c2c(CC)n[nH]c2)=O)(C)C)cc(C)cc(C)n1 CC1CC(COCC#N)CN(C(C2C=CC(=O)N=N2)=O)C1 N1(C(CCC(C)C)=O)CCC(CNC(c2nc3c(s2)CCCC3)=O)C(F)(F)CC1 CC(CCNC(c1cc2ccncc2[nH]1)=O)N=c1[nH]nc(C(F)F)s1 c1(OC)cc(CC(C)N(CC(c2ccccc2)O)C)ccn1 c1(NCC(c2cccc(C)c2)C)ccc(S(=O)(=O)NC2CCOC2)cc1Cl CCCC(C)(C)C(=O)NCCOCCC(=O)NCC1CCCC2(CC2)C1 N1(C(=O)C=CSc2ccccc2)CCC2CCN(C(=O)CSCC(F)(F)F)C2C1 c1(C(C(=O)NC2CC(C(=O)OCC)C2)(C)C)ccc2c(c1)OCO2 C1(=O)N=C2NN=C(S2)N1.CC(C(=O)OC(C)(C)C)C(C)n1cccn1 CC1CN(C(c2nccc(Cl)c2Cl)=O)C(C)CN1C(=O)C(C)C1CC1 c1(C(=O)NCC)cc2c(Cl)c(OC)ccc2[nH]1.C1(=O)C(C)(C)C2CCCN12 Cn1cc(C(=O)NCC2(O)CN(C(=O)CCOC3CCOC3)C2)c(=O)n(C)c1=O Cc1cccc(CN2CCN(C(=O)C(CO)c3ccccc3)C(C(C)C)C2)c1Br c1(C(=O)NC2CC(CCNC(c3n(CCC)cnc3)=O)C2)ccc(Cl)c(C)c1O C(N=c1nc2c(cnn2C)c(NCc2ccc(C)cc2F)[nH]1)C1CC(CC)C12CCC2 c1(OC)ccc(Cl)c(F)c1C(N1CCN(C(C2CSC2)=O)C(C(C)C)C1)=O Cc1ncnc(N(C(C)CCNC(c2ccccc2OCC(C)C)=O)C)c1Br C1(CNC(c2ccc(C(F)F)c(Cl)c2)=O)CC2(C1)CN(C(C13CCCC1C3)=O)C2 c1(OC)ccc(C(c2nnnn2C2CC2)NCC2C=CCC2)cc1C#N c1(NC(C2CN(C(c3ccc([N+](=O)[O-])o3)=O)CCC2O)=O)ccn2ncnc2c1 CC(C)C(CN(C)C)C(=O)NOONC=O.CC(F)F c1(C(N2CCC(Cc3ccccc3Cl)C2)=O)cc2ccccc2s1 c1(C(N2CCC(NC(=O)Cc3c(F)cccc3F)CC2)=O)cn2c(n1)COCC2 N1(C(C=Cc2ccc(C)o2)=O)CCC2C(C1)CN2C(C12CCC(C)(C1)OC2)=O CCC(CC)C(=O)NCC1CCC(CN(C(=O)COCCCF)C)CC1 C1(NC(C2(NC(C3CC(C)(CC)C3)=O)CC2(C)C)=O)CCCCCC1CO CC1CC(NC(c2cccn(C)c2=O)=O)CCN1c1nc(C(N)=O)ns1 C(C(CC(=O)N(C)OC1CCCCC1)OC)NC(c1cc(OC)no1)=O CN(C)S(=O)(=O)N(C)CC(=O)NCCCOCCNC(c1ccnc(O)c1)=O N12CC(CC1=O)NC2=O.C1(CC)CCC(NC(=O)CSCCC#N)CC1 C1(CC(=O)N(CCNC(c2cn(CC(=O)OC)nc2C)=O)CC)CCCC2(CCC2)O1 N(C(=NCC1CN(C)CCO1)NCc1nnc(C2CC2)s1)C(C1CCCC1)C#C C=CCC(C(=O)NC(c1ncc(C)[nH]1)C)NC(=O)Cc1ncccc1C N1(C(C(C)NS(CCC)(=O)=O)=O)CCC(CNC(=O)CC23CC(C2)C3)C(O)C1 CCCCC(O)C(=O)NC1CCCCCC1NC(=O)Cn1ccnn1 CC(C(=O)N(C)CC1(NC(=O)C(C)n2cccc2)CCC1)N(C)C(=O)C1CC1 Cc1[nH]nc(C(=O)N(C)CCN(C(c2cnn(CCO)c2C)=O)C(C)C)c1C C1(C)(C)CCCN1.C(F)(F)(C(F)(F)F)C1CCN(C(C2NCC(OC)C2)=O)C1 N1(C(C(=O)N(CCCCN(C)C)C)=O)CC(c2ccc(F)cc2)CC1(C)C c1(C(N2CCC(C(C)NC(=O)Cn3cccn3)CC2)=O)ccc(N)c(Cl)n1 Cc1ccc(NC(C2CN(C(=O)C(C)NC=O)C(C)(C)C2)=O)c(CO)c1 c1(NC(=O)NCC2C(OC)COC2)nn(-c2ccc(C)cc2)c2c1CCCC2 N12CC3CC1(C3)C(=O)NC(C)C2=O.CCCCCCOCC(=O)OCC C(c1ccc(F)cc1)=C(C)C(=O)NCC1CC(C)N(C(C2CCCCC2)=O)C1 N1(CC)CCOC(CC(=O)NCC(O)CN(C)C(c2ccc(SC)cc2)=O)C1 c12cnc(nc1O)C1(CCC1)N2.C1(NC)CC(=O)N(C2CCC2)C1 Cc1ccc2n[nH]cc2c1C(=O)NC(C)CC(C)NC(c1ccc(=N)[nH]c1)=O C1(CN(C(C2C(COC)(COC)C2)=O)C)CCCC(NC(c2sccc2F)=O)C1 C(=O)(C1CCCc2nncn21)NC1C(NC(c2c(C)nc(C(F)(F)F)o2)=O)CC1 c1(NC(C(N2C(CC)CC(O)C2)c2cc(Cl)ccn2)=O)cccc(Cl)c1C c1(C(=O)NC(C)CCNC(C2CCC2n2ccnc2)=O)cc(Cl)cc(F)c1N c1(C(=O)NCCC2CCN(C(C#CC3(C)CC3)=O)CC2)nccc2ccncc12 C(=O)(C(O)C(C(C)C)OCC)NCC1CCCN(C(C(C(=O)OCC)F)=O)C1 c1(CC)cccnc1C(=O)NCC(C)(C)CN(C(=O)CC1CC2CC2C1)C c1(N(C)CC2CC(O)C2)nc2ccccc2nc1N1CCCC2(CCCCO2)C1 C1(C(N2CCC(C(C)NC(CCNC(=O)NC)=O)C2)=O)CC2CCC(C1)N2C CC(C)CCC(C(=O)NCCC1(C)OCCO1)NC(C1CCC(C(N)=O)C1)=O c1(CC)nc(C(=O)NC2CCCC2CO)c2ccccn12.C(c1ccccc1)=CC Cc1cc(C)c(C(=O)NC2CC3(CCN(C(=O)CC4CCC4(F)F)C3)C2)c(C)c1 Cc1cc(C)n(C(C)C(N2CCC(C(C)NC(C3(C)CSC3)=O)CC2)=O)n1 C(C)(C(O)C(C)C)NC(C(c1occ(C(=O)OC)c1)OC)=O.C12CCC1C(=O)N2 c1(OC)ncc(C(=O)NCCN(C)C(c2[nH]nc(OC)c2Cl)=O)c(C)n1 N1(C(c2nc(COC)oc2)=O)CC(C(=O)NCCOC(=O)C2CC2)C2(CCC2)C1 CC(C)C(C(=O)N(C1CCN(C(C2CC3(CSC3)C2)=O)C1)C)C(C)C N1(C(CCOCCC)=O)CCC(CCNC(=O)CNS(=O)(=O)CC)C1 C(=O)(C(C)(C)CNC(=O)OC(=O)C1CC1)OCC c1(CNC(C(=O)Nc2ccc(OCC(=O)OC)c(Cl)c2)=O)n[nH]c2c1CCCC2 C1(NC(CCC2N(C)CCC2)=O)CCC2CC1CN2C(=O)CCc1cn[nH]c1 C1(F)(CNC(=O)CC2CC23CC3)CCC(CNC(c2ncoc2C2CC2)=O)C1 c1(NC2CCN(C(Cc3cc(C)cc(F)c3)=O)CC2C)ncnc2cccnc12 CCC(CC)CCCC(=O)N1CCC2(CC2C(=O)NCCc2cnco2)C1 CN1CCC(C(N2CCCC(c3nccs3)C2)C(=O)NCC(F)F)C1=O O=C(C1=NN(c2cccc(Cl)c2)C(=O)CC1)c1noc(C2CC2)n1 C(=O)(C(C)CC(F)(F)F)NCC1(CNC(C2CN(C(C)C)C2)=O)CC12CCC2 CCCCC(CC)CCC(=O)N(C)CC1CCCN(C(C2(CSC)CC2)=O)CC1 c1(CC(=O)NCC(CN(C(Cc2c(C)n[nH]c2)=O)C)C)cncc(Br)c1 c1(NC)cncc(C(=O)NC(C(=O)NCCCC(C)(F)F)C(C)O)c1 c1(C(N2C3C(CNC(c4ccc(SC)s4)=O)C(C3)C2)=O)ccnc2c1CCO2 C=CC(C)(O)CC(=O)NCC1C(C)CCCN1C(c1ccc(C)c(OC)c1)=O C#CC1(C(=O)NCC2CC(=O)N(C)C2)CCN(C(=O)C(C)N2CCCC2)C1 N1(C(c2cc(C(C)C)on2)=O)CCN(C(c2cc(CF)on2)=O)CC(C)(F)C1 c1(C(N2C(CCC)CN(C(=O)C3=CC(C)(C)C3)CC2)=O)cc(S(N)(=O)=O)sc1C c1(C(N(C2CN(C(C(CC)SC)=O)C2)C)=O)cc(OC(C)C)nc(Cl)c1 c1(OC)ccc(-n2nc(C3CCC(C)CC3)nc2CC2CC(C)C2)cc1 N#Cc1ccc(C(N2CC3CN(C(c4c(O)ccc(F)c4F)=O)C3C2)=O)cc1Cl Cc1c(F)cc(C(N2C3CCC2CN(C(C2(CC4CC4)CC2)=O)C3)=O)c(F)c1N c1(C(=O)OCCc2nc(C)on2)ccc(Br)c(Cl)c1 n1(CCNC(c2n(C)nnn2)(C)CC2CCCCC2)cccc(C2CC2)c1=O CC(CC(=O)NCC1(NC(=O)CC2CC(C)(C)OC2=O)CC1)C(F)F C12(C(N(CCC(=O)N(C)CC3CC4(CCC4)C3)CC=C)=O)CCC(OC)C1C2 c1(C(=O)NCCn2ccnc2)ccc(=NCc2ccc(C(F)F)nc2)[nH]c1 N1(C(C2(CC(C)C)CCNC2=O)=O)CCCCC(NC(=O)Cc2nccn2C)C1 N1(C(CNS(NC)(=O)=O)=O)CCN(C(C2COC(C)(C)CO2)=O)CC1CC1CC1 N1(C(c2n(CC)cnn2)=O)CC(NC(C2CCC(=O)N2)=O)CC12CCCCCC2 N1(C(C=CC(=O)OCC)=O)CC(C(C)O)(CNC(=O)CSCc2cccs2)C1 N1(C(C2C(C)=C2)=O)CC(C)CN(C(c2c(C)ccc3n[nH]cc23)=O)CC1C N1(C(C(CCSC)(C)C)=O)CCC(NC(C2Cc3ccccc3C2)=O)C(C)(C)C1 C(=O)(CN=S(C)(C)=O)NCC1CN(C(Cc2ncc(CC)[nH]2)=O)C(C)C1 C(=O)(C1=NOC(C)(C)C1)N1C(CNC(CCOCCN(C)C)=O)CC(O)C1 C#CCCN=c1scc(-c2sccc2C)n1C(C)CCOC C1(O)(CN(C(=O)CC(F)(F)Cl)C)CCCN(C(C2CC(=O)OC2(C)C)=O)C1 CCC(C)C(CC(=O)NCc1cc(=O)cc[nH]1)NC(=O)C(C)c1cccs1 c1(CC(N2C(Cn3cc(COC)nn3)CCC2)=O)c(F)cccc1Br c1(C(=O)NC2CN(C(c3ccnc(S)c3)=O)CCC2F)c[nH]c2nccc(Cl)c12 c1(OC)cc(Br)cnc1C(N1CC(NC(=O)CCCN(C)C)CC1CO)=O CCCC(C(=O)NCC(C1CC1)NC(c1cn(-c2ccccc2F)nn1)=O)OC C=CCCC(C(=O)NCC(=O)OC)NC(=O)N(C)C C1(COC)CN(C(=O)Cc2nccn2C)CCN1C(=O)Cn1cc(COC)nn1 c1(CC(=O)NCC2CC(COC)CN2C(C2CCOC2)=O)cc(C)cc(F)c1 C1(NC(c2c(CC)scn2)=O)CC2CC1N(C(c1cc(C(N)=O)cs1)=O)C2 c1(C(=O)NC2CC(C)(CC)N(C(=O)CC3CC=CC3)C2)cc(N)c(F)c(F)c1F c1(NC)cnc(C(C)C)nc1C(=O)NCC(C(C)C)NC(=O)CC1CCCCC1 CCC1=NOC(C(=O)NCC2CCC(C(=O)NC3CC3)CC2)C1.c12ccn-1n2 C(=O)(C(F)(F)Cn1cc(C)nn1)OC(C)(C)C.C1(Cc2nn[nH]n2)CC1(C)C CC1=NS(=O)(=O)NC=C1C(=O)NC1CC1NC(=O)C#CC(C)C N12CCC3CC3(CC1)C2=O.CC1C(=O)CCC1CSCNCCCC(=O)N(C)C CC(C)C(C(=O)N1CC(CO)(NC(=O)CC2CCC2)C1)n1cncn1 c1(OC)ccc(Cl)c(CN2CCCC(C)(C(=O)Nc3snc(C)c3C(N)=O)C2)c1 C1(=O)CCCCCn2cc(nn2)CCC2CN1C2.CCCCOC(C)=O N#CC1CCCC(CC(=O)N(C2CCOCC2)C2CCC2)C1.N(C1CC1)C=O N1(C(c2c(C)sc(O)n2)=O)CCC2(NC(C3CC3C3CCCCC3)=O)CCCC12 C=C1CCN(C(=O)Cc2cn(CC)nn2)C(C(=O)NC2CC(C)(O)C2)C1 c1(C(N2CCC(C(C)NC(c3csc(C(F)F)c3)=O)C2)=O)cn2ccnc2cn1 N1(C(C(CC(C)C)C)=O)CCc2[nH]nc(CNCC3(N4CCOCC4)CC3)c2C1 Cc1ccc(CC(=O)NC2CC3CN(C(c4ccoc4Br)=O)CC23)cc1[N+](=O)[O-] c1(C(=O)NCC(CNC(C(CSC)C)=O)CO)cc2c(nn1)CCC2 CC1CCN(C(=O)CC23CC(CNC(=O)CC4CCOC4)(C2)C3)CC1CO CC1C(NC(C2C=CCC2)=O)CC2CCC1N2C(=O)Cn1ncc2ccccc12 C12(C(=O)NCC3N(c4ccc(C)cc4)CCC3)CC3CC(CC(C3)C1N)C2 c1(CC(=O)NC2CCC(CNC(C3CC=CCC3)=O)C2)ccnc(O)c1 C1(OC(C)C(=O)NC2CCCCN2C(=O)OC(C)(C)C)CCC2(CC1)CC2 N1(C(c2[nH]c(=NC)sc2)=O)CC2(C1)CN(C(c1ccccc1C(C)(C)C)=O)C2 c1(C(N(C2CCC(NC(C3(OC)CCOC3)=O)CC2)C)=O)nccc(C#N)c1F c12ocnc1C(=O)N2.C(C)(C(=O)NC1CC(=C2CC2)C1)SCCC N1(C(C(C(C)C)SC)=O)CCCC(C)(CNC(=O)C=Cc2ccccc2)C1 c1(C(=O)NC(CN(C(CCOCC#C)=O)C)(C)C)ccc(C#N)nc1O N1(C(C(C)NS(CC)(=O)=O)=O)CC(N(C)C(c2ccc(COC)nc2)=O)C(O)C1 C(=O)(CC(C)(C1CC1)C1CC1)N.C(C(=O)NC(CCCN(C)C)C1CC1)N(C)C C1(C(N2CC(O)(CNC(C(CC)O)=O)C2)=O)COc2ccc(OC)cc2C1 O=C(C1=NN2CCCN=C2N1)NCC1CCCN(C(=O)C2=COCC2)C1 C1(C(=O)NCC2CC3CC3C2)(COC)CN(C(=O)CN(C)C(C)=O)C1 CCCC(O)C(=O)NC(CNC(c1[nH]cc(C)c1C)=O)C(C)(C)C C1(C(N)=O)CNC(=O)CN1C(=O)C1=NOC(CNC(=O)Cn2c(O)nnc2O)C1 CCC(C)C(O)C(=O)NC1(CNC(c2cccc(CF)c2)=O)CCOCC1 N1(C(C2CCN(C(C(CC(C)C)O)=O)C2(C)C)=O)CCOC2(CCC2)C1 C(=O)(CC1=NNC(=O)C1)N1CCC2(NC(CC(C)(C)n3cc(CO)nn3)=O)C(C1)C2 C(=O)(CC1=CCOCC1)NCC12C(CN(C(c3cc(CC)nc(O)c3)=O)C1)C2 C=CC(C)(CCOC)C(=O)NCC#CC(=O)NCc1sc(C)cc1C C(C(O)CC(=O)N(C1CN(C(c2ccncc2C(F)F)=O)C1)C)N(C)C N1(CC(=O)NC2CCCC(CC(=O)NCCCC3C(C)C3)C2)C(=O)CCCC1=O N1(C(CCCOCCC)=O)CCC(CNC(=O)CC2CCSCC2)C(CC)C1 C(=O)(C(F)CCC(C)C)N1C2CC(CNC(CCN(CC)CC)=O)(OC2)C1 c1(CNC(CCOc2cccc(C(C)C)c2)=O)cc(F)cc(Br)c1O CC(C)CC(CCc1ccccc1)C(=O)NCC1CCCCN1C(=O)C(C)(F)F C1(F)(C(N2CCC(N(C(C(F)=CCC)=O)CC)CC2)=O)CCN(C)CC1 N1(C(=O)Nc2ccc(C)cn2)CC(NC2CCC(C)(C)OC2)CC(C)C1 c1(C(N2CC(CCCNC(c3c(CC)noc3)=O)OCC2)=O)ccc(F)cc1O N1(C(C2(CC)CCCC2)=O)CC2CCN(C(c3cc(F)c(N)cc3F)=O)CC2C1 c1(C(N(C)CC=CC(=O)NCC2COCCO2)=O)cccc(CO)c1 C1(C(=O)NCCC(C)N(CCC)C)C2CC(O)C(C2)N1C(C1(C2CC2)CCC1)=O c1(C(=O)NC(C2CCOC2)COC)cc2cccc(-c3ccc(B(O)O)cc3)c2[nH]1 N1(C(C(C2CC2)SC)=O)C2CCCC1CN(C(C1CCC3(CCC3)O1)=O)C2 C(=O)(CCCCCCCS(C)(=O)=O)NCC1(F)CN(C(C2C(C=C)C2)=O)C1 Cc1ccc(O)cc1NC(=O)C(CC1CCCC1)NC(=O)CCc1ccoc1 [N-]=[N+]=NCCCCC(=O)N1CC=CC1CSC.[nH]1cc(C(O)CC)nn1 c1(C(N2CC(C(=O)NC3CC(CC)C3)C(O)C2)=O)ccc2c(c1)CCC(=O)N2 Cn1cc(Cl)cc1C(N1CC(CNC(c2cccc(CC3CC3)n2)=O)C(O)C1)=O Cc1c(N)cc(C(N2CCCC(F)(CNC(C3CC=CCC3)=O)CC2)=O)cc1N c1(C(=O)NC2C3CN(C(c4c(C)[nH][nH]c4=N)=O)C(C3)C2)sc2ncccc2c1Cl C(=O)(C1(C)CCCc2ccccc21)NC1CN(C(c2cc(C)[nH]c2C)=O)CC1C C(N=c1ccnc(C2CC2)[nH]1)C1N(C(c2cc(Cl)ncc2F)=O)CCC1 N1(C(C2CCC(OCC)CC2)=O)CCN(C(=O)CC(C)(C)OC)CC1CF N1(C(C(CC)(C)F)=O)CC2CC(C)N(C(c3cccc4ncnn34)=O)C2C1 CN=c1[nH]cc(C(=O)NCC2CN(C(=O)C3=CCC3)CC2C)o1 CON=CC(=O)N(C)CC1CC(C)N1C(=O)OC(C)(C)C CC1(C)COC(CCCNC2CC(CF)C2)C1.C1(C(=O)O)CCC1 C1(NC(c2cc(SC)c(C)o2)=O)CC(F)CN(C(c2nnc(C(C)(C)C)s2)=O)C1 C1(C2(C)CC2)CN(C(=O)Cc2cn(C)cn2)CCN1C(=O)CN=[N+]=[N-] Cc1nn[nH]c1C(N1CC(O)(C(C)NC(c2cn(CCF)nn2)=O)C1)=O c1(C(N(C2CC2)CC2N(C(c3n(C)cnc3)=O)CCC2)=O)cnc2n1CCS2 C1(N(C(CN(CC)CC)=O)C)CC2CC1N(C(=O)C(c1cccnc1)C)C2 c1(C(=O)NCCCC(C)NC(c2cc(-c3ccco3)no2)=O)sccc1C#N CN1CCCC12CCN(C(=O)C1=CCCN(C(C3C4CCC(F)C34)=O)C1)C2 C(=O)(CCCCCNC(C1(CCN(C)C)CC1)=O)ON.CC1(C)CN1 C=CC1(CC(=O)NCCSC)CN(C(=O)C(CO)c2ccccc2)C1 C1(CN(C(CCOC(C)C)=O)C)CN(C(=O)CC(=O)NC2CC2)CCO1 C1(C(=O)NCCc2cc[nH]n2)CN(C(=O)CCC2CC2CC2CC2)CC12CCC2 C(CCC(=O)NCC=CCC(=O)NCCC1(C)CCCO1)N(C)C C(=O)(C(C(C)C)NC(C)=O)NC(CCCNC(c1ccc(SCCC)o1)=O)C CCCS(=O)(=O)c1ccc(C(=O)NCCN(C(=O)CCc2ncc[nH]2)CC)cc1 C(CN=c1cnc(NCC(CC)(CO)N2CCOCC2)c[nH]1)OCC C(=O)(C(CN(c1ccccc1)C)NC(=O)NCC1CC(CO)C1)OC N1(CC(C2CCOCC2)CN)CCc2c(cccc2S(N)(=O)=O)C1 N1(Cc2ncc(OC)nc2)CCC(F)(F)C(C(=O)NC2CCN(C)CC2)C1 c1(C(N2CCC3(C2)CN(C(C2CC2Br)=O)C3)=O)ccc2c[nH]nc2n1 N#Cc1ccc(CNC(=O)C(C2CC2)NC(=O)CNc2cccnc2)o1 N1(C(CC)C)C(=O)NC(c2cn(C3CCCC3)nn2)C2=C1C(C)(C)NC2=O C1(C(N2CC(CCn3cc(CCC(C)O)nn3)C2)=O)COc2cc(Cl)ccc2O1 c1(C(N2CCC(C)(NC(C=CCC)=O)C2)=O)c[nH]c2ccc(Cl)cc2c1=O c1(N(c2nccc(N)n2)C(C2CCCNC2)OC)ccc(F)c(Br)c1F.CO N1(C(C2(C)CCC2)=O)CCCN(C(c2ccc(Br)c(Cl)c2)=O)C(CO)C1 c1(CCCNC(C(n2cc(C(CC)OC)nn2)C)=O)cccc(C)c1 Cc1ccc2c(c1)SC(C(=O)NCC1CC1NC(c1sccc1S(C)(=O)=O)=O)C2 c1(C(=O)NCC2(C)CCCN(C(C3(O)CC3)=O)C2)cnc2ncc(Cl)cn12 c1(C(=O)NCC(CN(C(C(CSC)C)=O)C)O)cc(C)nc2c1CCCC2 c1(C(=O)NCC2CC(NC(C3(CC=C)CCCOC3)=O)C2)cc(C)cc(F)c1 c1(C(c2n(CCCOC)nnn2)NC(c2ncc(Br)s2)C)sc(Br)nc1Cl c1(OC)cc(C(=O)NCC2CN(c3cc(O)ncn3)CCO2)ccc1C#N C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)C1CCN(C(c2ccc(C)cc2Cl)=O)C1 N1(C(C(CC(C)C)C)=O)CCCN(C(c2ccc3c(c2)CCC3)=O)C(C)C1 CC1(C)CCC(C)(C(=O)NC2CC3(NC(c4cnsc4)=O)COC2C3)CC1 c1(CN(c2n(C3CCC(C(=O)OC)C3)nnn2)CC(=C)C)cc2occc2s1 C(=O)(C(C(C)(C)C)NC(c1cn(C2CC2)cn1)=O)N(C)Cc1c[nH]nc1CO CC1(C)COCC1CC(=O)NCC1CC(NC(=O)C=Cc2cccnc2)C1 C1(CCNC(C(CO)N(C)C)=O)CCN(C(C2(CF)CCOCC2)=O)CC1(F)F c1(CNC(CC2(C)CC2(F)Cl)=O)cccc2c1CCN(C(C1CC13CC3)=O)C2 c1(C(N(C)CC2N(C(CCC)=O)CCC2)=O)cnc(OC)c(C)c1 C(=O)(C(O)CC[S+](C)C)N1CCC(C)(CNC(c2c(C)cccc2)=O)C1 N1(C(C(CCSC)(C)C)=O)CCC(C2CCN(C(C3CCCO3)=O)CC2)CC1 C1(NC(C(C)O)=O)CCC2(CC1)CC2Nc1cc(O)nc(=O)n1C c1(C(N(C(C)CC2CC2)C)=O)coc2c1CN(C(C13CCC(C)(C1)OC3)=O)C2 c1(CNc2ccc(N3CCC(N)CC3)cc2)cc2ccccc2nc1Cl N1(C(c2c(OC)cnnc2)=O)CCOCCC1C(=O)NC1(c2ccsc2)CC1 Cc1c(Cl)ccc(C(=O)NC2CN(C(=O)CNC(=O)CN(C)C)CC2(C)C)c1O CC1(C)CN(C(C2(CF)CC(F)(F)C2)=O)CC1CNC(=O)Cn1cccnc1=O C1(C(N2C3CC(CNC(=O)CCCC4CCC4)C2CC3)=O)CCc2nncn2C1 CS(=O)(=O)c1ccc(C=CC(=O)NC2CCC2NC(c2cccc(N)c2F)=O)o1 c1(C(=O)NC2C(NC(c3ccc(C)o3)=O)CC2)c(C2CC2)noc1C c1(C(C(=O)NCC(CC)(C)NC(=O)CC(C)CF)(C)C)c(F)cccc1F Cc1nn(C)c2sc(C(=O)N(C3CC4CC3N(C(c3ccns3)=O)C4)C)cc12 c1(C(=O)NC2C(NC(C(n3cc(C)nc3)(C)C)=O)COC2)ccc2scnc2c1 c1(CCN(CC(F)(F)F)C(C2CC(=O)N(O)C2)=O)ccc(Cl)cc1 CC1(C)CN(C(C2CN(CP(C)(C)=O)C2)=O)CC2(CN(C(=O)C(O)C3CC3)C2)O1 N1(C(c2ccc(CC)[nH]2)=O)CCCC(CC(=O)N(C2CC2(C)C)C)CC1 C(N=c1[nH]cc2ncnc-2[nH]1)C1C(C)CN(C(c2cc[n+]([O-])cc2)=O)C1 c1(C(=O)NC(C(C)NC(c2n(OC)cnc2C)=O)C(C)C)cnn2cccnc12 N1(C(c2c(C)n(C)cc2)=O)CC2(CCC2NC(=O)CNC(c2cccnc2)=O)C1 C1(OCC)CN(C(c2cc(C(F)F)nn2C)=O)CC1CNC(=O)C(C)=C1CC1 C12(CNC(c3ccccn3)=O)CCC1CN(C(c1cccs1)=O)C2 C1(C(=O)NCCc2cn(-c3cc(C(=O)OC)ncc3)nn2)CCC12CCOCC2 N1(C(C(C)OCCOC)=O)CC2(CC(NC(=O)C=CC3CCCC3)CO2)C1 C12(NC(C(C)SC(F)(F)F)=O)CCCC(NC(c3ccc(C(C)F)cc3)=O)(C1)C2 S(=O)(=O)(c1ccc2[nH]c(=NC(C)COC)sc2c1)N1CCN(CCOC)CC1 c1(N(C2CCN(C(C34CCC3CC4)=O)C2)C(=O)CSC)cccc(C)c1 C1(NC(=O)CCc2ccc(O)cc2)CCSC12CN(C(c1csc(O)n1)=O)C2 CC(c1ccccc1C)=CC(=O)NCCCCNC(=O)CC1CC2CC2C1 c1(C(CC)NC(c2sc(NC(C3COCCO3)=O)nc2C)=O)cc(F)cc(F)c1 c1(C(N(C2CCCC2)CCNC(c2cnc(SC)s2)=O)=O)cccc(Cl)c1 c1(Cn2c(COCC)ncc2)c(Br)cc(C(=O)O)n1C CCCC(C)CC(=O)N1CCCC1C(=O)N(C1CCN(OC)CC1)C C1(NC(c2ccc(C#N)cc2)=O)CN(C(c2cnc[nH]2)=O)C2(CCCOC2)C1 c1(C(c2n(CCCSC)nnn2)NC2(C3CC3)CC2)ccc(OC(C)C)cc1 N1(C(C2=CCCC2C)=O)CCCC2(CCC(NC(c3cc(Cl)ccn3)=O)C2)C1 C1(O)(C(=O)Nc2ccc(O)cc2)CCN(CC2(CC)CCNC2)CC1 c1(N2CCC(C)(C(=O)NC)C2)cc(N2CCNC(=O)CC2)nc(COC)n1 C1(NC(c2cc(-c3ccco3)[nH]n2)=O)C2CCC1N(C(C1(F)CC=CCC1)=O)C2 C=CCC(CC(C)C)C(=O)NCC1CN(C(=O)CN(C)C(N)=O)CCO1 C(=O)(C1=CCCOCC1)N1C(C(=O)NCC2(C#N)CC2)CC(O)C1 C1(CC(=O)NCC(CCCC)NC(c2nc(C)oc2C)=O)CC(O)C12CCC2 C(CCCCCNC(C1(F)CC=CC1)=O)N(C(=O)CC1CCOC1)C N1(C(C(C)OCC#C)=O)CCC(C)N(C(c2cn(CC(N)=O)nn2)=O)CC1 C1(NC(C(C2CC2)OC)=O)CCN(C(c2ccc(F)cc2Cl)=O)C(C)C1 CCCC(C(=O)NC1CCC1)NC(C1(C)COC(=O)N1)=O CCCC(CCC)CC(=O)NC1CCCC1NC(=O)CC1CCC(=O)O1 Cc1cc(C(=O)NCc2cc(C(=O)NCC3CCC(C(N)=O)O3)cs2)c(C)n1C N1(C(c2c(C)n[nH]c2)=O)CCC2(CC1)CC(CNC(=O)C1CCc3c[nH]nc31)C2 c1(N(c2cccc(CC)c2O)CCC2CCC2)ncnc2n[nH]c(I)c12 C1(C(=O)NC23C(CN(C(C)=O)C2)C3)CC2CSCC(C1)C2(F)F N1(C(c2ccn(CCN3CCN(C)CC3)n2)=O)CC=CC(C(=O)OC)C1 C1(C)(CNC(C(C(C)(C)O)F)=O)CC(F)(F)CN1C(=O)Cn1nc(O)ccc1=O N1(C(C(CCOC)C)=O)CCC(C)(C)C(CNC(C2(O)CCCCC2)=O)C1 C1(C(N2CCC(C#C)(O)C2)=O)CC(O)C(O)CC1CNC(=O)C(C)(C)CC#N C1(CC)CCCCC1C(=O)NCc1nc(CNC(=O)C(C)SC(C)C)cs1 c1(C(N(CCC2CCC2)CC)=O)nc(-c2ccncc2)nc2ccc(OC)cc12 CC1CCC(C)(C(=O)NC(C)C(CO)NC(c2scnc2C2CC2)=O)CC1 c1(C(=O)NCC2(NC3C(=O)NCCC3C)CC(=C)C2)ccc2[nH]ccc2c1 c1(C(=O)OC)c(CNC(c2ccccc2F)c2ccco2)ccn1C n1(CC(=O)NC23CC(CNC(C(C)CO)=O)(OC2)C3)nnc2ccccc2c1=O c1(OC)cc(C(=O)NCC23CCC(CC2)N3C(=O)Cn2cnnc2O)cc(Cl)n1 c1(OC(C)C(=O)NC2CC(C(C)(C)O)C2)ccc(F)cc1F C1(CNC(C(C)OCCC=C)=O)CCC2(CCN(C(=O)C(F)=CC3CC3)CC2)O1 Nc1c(C(N2CCCC3(C2)CN(C(=O)CCCF)C3)=O)sc2ncccc12 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C(C)C)CNC(C1CCOC1C1CC1)=O N1(C2CCN(C(N(C3C(C)OC(C)C3C)C)=O)CC2)C(=O)c2ccccc2C1=O C1(CNC(c2csnn2)=O)CN(C(c2ccc3ccoc3c2)=O)C2CCN1C2 Cn1nc(C(=O)NCCc2n[nH]cc2C(=O)NCCc2nc(CO)no2)cc1F c1(C(=O)NC2CN(C(CC(C=C)C)=O)CC(F)C2)cnn2ccc(Cl)c(F)c12 c1(OC)cc(C(N2CCC(c3ccc(F)cc3F)CC2)=O)cc(F)c1C#N c1(C(=O)NCC2CC(NC(C3OCCC(C)C3)=O)C2)nnn2c1CSCC2 C#Cc1ccc(C(=O)NC2CC(NC(C3CC3C(C)(F)F)=O)C2)cc1C C1(C(N(CC(C)NC(C2(O)CCSC2)=O)C)=O)CC(C)(C)OC(C)(C)C1 Cc1c(C(=O)NCC23CC2CN(C(c2cc(C4CC4)nn2C)=O)C3)ncn1C CC1CC2CCC(C1)N2C(C1CCOC1CNC(c1ccc(O)cc1)=O)=O C(c1ccc(C)c(C)c1)=CC(=O)NCC1CCC(NC(c2cnc(OC)s2)=O)C1 C(=O)(CS(=O)(=O)CCCc1ccccc1)NCC1CN(C(C(CC=C)C)=O)CC1O C1(C)(CNC(c2c(C)scn2)=O)CCCN(c2cc(Cl)nc(C(C)(C)C)n2)C1 C(C)(C)(CCCC(=O)N(C1CCCC(O)C1)C)NC(C(C)OC)=O C1(C(N(CCCNC(=O)CNC(C2CCC2)=O)C)=O)C2COCC12 c1(CC(=O)NC2(CNC(C3N(C)C(=O)NC3)=O)CCCC2)cccc2ccsc12 C(C)(CCC(=O)N1CCCC(NC(c2cncn2C2CC2)=O)C1)OCC C(=O)(C(F)CC(C)(C)NC(c1c[nH]c(=N)o1)=O)N1C(C)CS(=O)CC1 NS(=O)(=O)c1cc(C(N2CC3CC2CN3C(=O)Cc2ncc(Cl)s2)=O)cs1 N1(C(C2C=C(C)CS2)=O)CC=CCC1C(=O)N(CC(O)C1CC1)C C1(CC=C)(NC(=O)CC(C)(F)F)CCN(C(C2CC3CC2CC3O)=O)CC1 N1(C(C2(CCC)CC2)=O)CC2CCC(C1)N2C(=O)C(O)C1CC1 C1(F)(C(=O)NCCC=CC=C)CCN(C(=O)C(CC)SC)CC1 c1(C(N2C(CO)CC(NC(C3C(C)C3)=O)C2)=O)ccc2c(c1)N(C)C(=O)CO2 NS(=O)(=O)CC(=O)N1CC(CO)(NC(=O)C=CC(F)(F)F)C1 N(C(=NCCC(C)SC)NC(c1ccccc1OC)C)Cc1cc(CC)no1 c1(C(C)C)ccc(O)c(C(N2CCC(NC(C3CC(CF)C3)=O)C2)=O)c1 S(=O)(=O)(c1ccc(N2CC3CCC(C2)O3)c2cnccc12)NCCC#N Cc1csc(=O)n1CC(c1c(-c2cn(C(C(C(C)C)N(C)C)C)nn2)cncn1)=O CCC(CC(F)F)C(=O)NC1(C)CN(C(c2ccc(OC(F)F)c(Cl)c2)=O)C1 N1(C(c2nn(CC)c(O)c2)=O)CCC(C2CCN(C(=O)CC(C)(C)N(C)C)C2)C1 C1(CC(N)=O)(NC(CCOC)=O)CCCN(C(c2cc(C)n(C(C)C)c2C)=O)C1 C1(C(N2CC(N(CC=C)C)C2)=O)C(CNC(c2nnsc2C)=O)C1(C)C N1(C(CC=C)=O)CCCC(C(N2CC(C(N)=O)C(CCC)C2)=O)CC1 C1(C(=O)NC2(CF)CCN(C(CCOC)=O)C2)CC2CC1CC2(F)F C1(C(N2CC(N(C(=O)Cc3cnco3)C)C2)=O)CCCC2C1C2(F)F CC1CC(NC(c2nnc(S)n2C)=O)CN(C(c2ccn(C)c(=O)c2)=O)C1 c1(C(N(CC(CC)NC(c2conc2C(C)C)=O)C)=O)ccc(OC)cc1C c1(SCC(=O)NCCC(O)CNC(C2(CO)CC2)=O)ccccc1F C1(NC(c2ccn(C)c2)=O)COCCN(C(c2n[nH]c(C3CC3)n2)=O)C1 c1(CN(C(c2c[nH]cc2CC)C(=O)NCCOCC)CCO)cccc(F)c1C c1(CNC(C2CC23CCNC3)=O)c(F)cccc1Br C(=O)(CC(C(F)F)c1ccccc1F)NC1C(NC(C2(CC=C)CCC2)=O)C1 C1(C(=O)NCc2ccccc2)CC(=O)N(CCN(C(C2C3COCC23)=O)CC)C1 N1(C(c2ccc(=N)[nH]c2)=O)CC2(CC2)CC1CNC(C1CCCO1)=O CC(C)(CC(=O)NC1CCC1NC(c1cc[nH]c1)=O)C(F)F C[S+](C)CCC(O)C(=O)NC1CN(C(c2coc(C(F)F)n2)=O)CCC1F Cc1nc(C2CC2)sc1C(=O)NCC12CC1CN(C(=O)CCC(F)F)C2 c1(CN(CCNC(c2nn[nH]n2)=O)CC)nc(Br)ccc1OC C1(C)(NC(C(CC)=CC)=O)CCN(C(c2sc(C(F)(F)F)nc2C)=O)C1 Cc1cc(O)cc(=O)n1C(C)C(=O)NCCC1COCCN1C(=O)C=C1CCC1 c1(C(=O)NCC(CC)NC(C2COC(C)C2)=O)cc(F)cc(N)c1N c1(CC)noc(C)c1C(=O)NC1C2CC1N(C(c1ccnn1CCF)=O)C2 C1(OC)CC2CC(C(N3CCCC3CNC(=O)C(C)(C)C3CCOCC3)=O)CC12 N1(C(c2cnc(OC)nc2C)=O)CC(C)CN(C(C2CCC3CC3C2)=O)C(C)C1 c1(C(N(C(C)CNC(=O)C=CC2CCCC2)C)=O)ccnc2ncccc12 c1(OC)cccc(CC(=O)NC(C)CC2CN(C(=O)C(C)(C)N(C)C)C2)c1 C1(NC(=O)C=Cc2ccccn2)CN(C(C2SCCCS2)=O)CC12CC2 C1(C)(CCC)CCN(C(=O)C(CCOCCO)NC(C2COCCC2C)=O)C1 N1(C(c2[nH]cc(C)c2C)=O)CCN(C(=O)CSCCC(C)C)C2(CC2)C1 N1(CC(=O)NC23CCN(C(=O)CCCC4CC4)CC2C3)CCCCCCC1=O C1(C(=O)NC2(C)CCN(C(COC(C)(C)C)=O)C2)CCc2nnc(O)n2C1 Cc1cc(=NCC2CCCC2NC(C23CCCC(C2)OC3)=O)c([N+](=O)[O-])c(C)[nH]1 N1(C(CCCc2c(C)ccs2)=O)CCC(NC(=O)C=CS(C)(=O)=O)C(CO)CC1 CCCC(O)(CNC1CCCC1CCC)C(F)(F)F c1(OC)cc(F)cc(CN2CCC(O)C2C(=O)Nc2ccc(F)cc2O)c1Br C12(NC(c3cc(C)cc(N)c3)=O)CCCC1CN(C(=O)Cn1c(C)csc1=O)C2 N1(C(C=C(C)Cl)=O)CCC2(CCC2)C(NC(=O)C(CCC(N)=O)NC(N)=O)C1 CC12CCN(C(=O)CC3CCSCC3)C1CN(C(c1ccc(C3CC3)cn1)=O)C2 c1(C(=O)NC(CC=C)C(=O)N2CCOC(CC(C)C)C2)c[nH]c2ccncc12 c1(CCCC(=O)NCC(CCOC)NC(=O)C(C)C2CCC2)ccc(F)cc1 O=C1NC2CN(C(=O)CC3C=CS(=O)(=O)C3)CC2N1 N1(C(C2C(CC)C2)=O)CC(COC)CC1CNC(c1sc(C)cc1C)=O N1(C(c2n(CC)ncc2)=O)CCC(NC(=O)CSCC(C)(C)C)C1C1CC1 N1(C(CCCSC)=O)CCC(C)(C)C(C(=O)NCC2CCC3(CC3)C2)C1 Cc1nc(Cl)[nH]c(=NC2CC3CCCC(C2)N3C(C2CCC3(CC2)CC3)=O)c1F C(=O)(CS(=O)(=O)N1CC(O)CC1C(=O)NCc1ccncc1Cl)OC N1(C(C(CCC)C)=O)CCC2C(CCCN2C(=O)CCc2ncc(C)[nH]2)C1 Cc1ccc(CC(=O)NC2CC2NC(c2cc(C(F)F)cs2)=O)o1 C(C(C)(CO)NC(C1CSCN1C(=O)Cc1ccoc1C)=O)NC(C=CCC)=O c1(C(=O)NC2CN(C(=O)Cn3ccc(C4CC4)n3)C2)ccc(-c2cc[nH]n2)cc1 N1(C(C(=Cc2cnc[nH]2)C)=O)CCCC(C2(NC(C3CSCCS3)=O)CC2)C1 c1(C(=O)NC(c2c(C)cccc2Cl)C)nc2n(c1Cl)CCCC2 C1(C(=O)NOCCC(F)F)CC(O)CCN1C(=O)C(O)C1CCCC1 Cc1nc(Cl)ccc1C(=O)NC1CCN(C(=O)C(C)CN(C)C)CC1C CC12CC(C(=O)NC3CC(NC(=O)C(C)(C)c4ccccc4)CC3O)(CCO1)C2 c1(CNC(NOCC(CCCC)O)=O)nc(Br)ccc1OC c1(NC)cccc(C(N2CCC(CF)(NC(c3ccc[n+]([O-])c3)=O)C2)=O)n1 C1(c2nnnn2C(c2nnc(C)s2)C)(NCC2CC(OCC)C2)CCCSC1 c1(OCC(=O)NC2CC2CNC(c2cccnc2)=O)ccccc1 CCC(C#N)(CC)C(=O)N1CCC(O)C(NC(=O)CCn2cccn2)C1 N1(C(C(C)Oc2cccc(OCC(C)C)c2)=O)CCc2sccc2C1 Cc1cc(C(N2CCCCC2CCNC(=O)C(O)C(C)(C)C)=O)cnc1C(F)F C12(C(=O)NCC(O)C3(Cl)CC3)CCC(CN(C(C3(O)CCSCC3)=O)C1)C2 C1(C(N(CCC(=O)N(C)CC)C)=O)CCCC1O.O(C(F)F)CCO C1(OC)CC(C(=O)NC(=O)CC2C=CCCC2)CN(C(c2ccc(F)cc2C)=O)C1 N1(C(C2C(C)CCN2C(=O)C=Cc2cccnc2)=O)CCCC(C#N)C1 C1(C2CN(C(c3cccc(C#C)c3)=O)C2)(NC(C(CC#C)C)=O)CC1 c1(C(=O)NC(C(C(C)C)NC(c2c(C)cc(=N)[nH]c2)=O)C)cc(Cl)c(F)cc1F CCC(CCC(=O)NCC1CC2CCC1N2C(=O)CCc1cccc(C)c1)OC C1(C(N2CC(CN(C(=O)C(F)C3CCOC3)C)C2)=O)C2CCC1(C)C2(C)C CC1(C)CCCC1C(N1CCCCC1CCNC(c1ccn(CCF)n1)=O)=O Cc1c(F)ccc(C(=O)NC2CCN(C(=O)CCc3cnn[nH]3)CC2C)c1N c1(C(N2CCC(NC(CC=CC)=O)C(CC)C2)=O)n[nH]c2ccc(O)cc12 CCCC(C)(CC)C(=O)N1CC2CC1C2NC(=O)C(O)CCCC c1(SC)cnc(N2CCOCC2CNC(=O)CCc2cncnc2)nc1 c1(C(=O)OCC)nc(C)cc(=NC2CCCC2C(C)NCCOCCN(C)C)[nH]1 CC1CCC(C)(C(=O)NC2CN(C(=O)CN(S(=O)(=O)CCOCCOC)C)C2)C1 C1(NC(c2c(C)nsc2)=O)CN(C(=O)CN(C)CCO)CC1O Cc1cccc2c1OC(C(=O)NCC1CC(O)CN1C(c1cc(Br)co1)=O)C2 C1(NC(C=C(CC)CC)=O)CN(C(=O)CCC(=O)Nc2nccs2)CCC1F c1(N2CCCC(C(=O)NC(CSCC)=O)CC2)nc(CC)nc2ccccc12 C(=O)C1=CC2(CCN(C(C)=O)C2)C1.N1(CC(NOC(C)C)=O)CCN(C)CC1 N1(C(CCCC(C)(C)NC(C2CC3(CC(=O)C3)C2)=O)=O)CCC(C2CCOC2)C1 C(=O)(CCCCCCNC(c1ccc(N)cn1)=O)NC1(C#C)CC1 C(=O)(C1CCCn2ncnc21)N1CC(O)(CCCNC(c2cccc(C)n2)=O)C1 N1(C(CC(C)(C)C)=O)CC2CC1CC2NC(=O)Cc1ccc(F)cc1 C1(CNC(c2c(C)nn(CC)c2C)=O)C2CCCC1N(C(=O)CCC1(C)N=N1)C2 c1(C(=O)OC)nc(CN(C(=O)C(C2CC(F)(F)C2)Oc2ccccc2)CC)oc1C C1(C(c2nnnn2CC2CC2)NCC(C)C2CCC2)C2(CCC2)C12CCC2 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCN(C(CC(C=C)C)=O)CC12CCC2 N1(C(CCCCC#C)=O)CCOCC(C)(CNC(=O)C2=CCC2)C1 C1(CNC(c2ccc(C=C)cc2)=O)CC2COCC2N1C(C1CCN1CC)=O C1(CCOC)(NC(=O)CC2CC(C)C2)CCN(C(C2CCCC(F)(F)C2)=O)CC1 C(CCCCC(=O)NCC1CCCC1NC(=O)OC(C)(C)C)N(C(=O)C(C)(F)F)C C(=O)(C(C)C(O)CC(C)C)NCC1(C(N2CC(C)OC(C)(C)C2)=O)CC(C)(C)C1 c1(CCC)nnc(S)n1CC(=O)NC1CN(C(=O)C=Cc2cnc[nH]2)C1 C1(NC(CC2N(C(C3CC(CC)C3)=O)CCCC2)=O)CC2CC1C(O)C2O c1(C(N2CC(NC(c3ccccc3)=O)C3(C2)CC3)=O)ccnc2cc(F)cnc12 c1(C(N(C(C)CNC(=O)C(O)C2CC2)C)=O)ccnc(C(F)(F)F)c1F c1(OCC)ccc(C(=O)NCC(C(C)(C)C)NC(c2cnc(S)n2C)=O)cc1 Oc1cc(CCn2cc(-c3c(Cl)cncc3Cl)nn2)ccc1Br c1(OCCCNC(c2n(CCCC(=O)OC)nnn2)C(C)C)ccc(Br)cc1 C1(CNC(C(F)OC)=O)CCC(CNC(=O)CCc2ccc(F)nc2)CC1 C1(CN(c2ccnc(N(C)Cc3nnc(Br)n3C)n2)C)CCCC(O)C1 c12ccccc1CC(C)C(=O)N2.C(C(C)CN(C)C)N(C(C=C(C)Cl)=O)C N1(C(c2cc(Cl)c(OC)c(Cl)c2)=O)CCc2sc(-c3c(C)noc3C)cc2C1 N1(C(CC(C)C2CC2)=O)CC2(CCN(C(=O)CC3COC(C)(C)CO3)C2)C1 C1(CNC(C(C#C)(C)C)=O)CN(C(c2[nH]c(O)nc2C)=O)CC1(C)C C1(NC(CCC2CCC(=O)N2)=O)CCCCN(C(C2CCSC2)=O)C1 C1(NC(C(C)=CC)=O)CN(C(C2C3CCC4C(C3)CC24)=O)Cc2nccn2C1 C1(c2cn(C)nc2)CCCN1N1CCC(CCNC(=O)OC(C)(C)C)C1 C1(O)(C(N2CCN(C(CC)=O)C(CC)C2)=O)CCCC(C)(C)C1 CCC(CC)C(C)C(=O)N(C1CCCCC1NC(c1occ2c1CCOC2)=O)C C1(NC(c2ccc(C(=O)OC)cc2)=O)(CO)CC2(CCC2)C1 C1(NC(C(C(C)O)(C)C)=O)CCCCCCC1NC(=O)C=C1CCCCC1 C1(NC(CCOC)=O)CC2CC1N(C(c1nnn(-c3ccc(F)cc3)c1C)=O)C2 c1(OC(C)C)cccc(-c2cn(C(C)CC3CCN(C(=O)CO)CC3)nn2)c1F c1(OC)ccc2ccc(C(=O)OCCC3CN(C(=O)CCF)CC(C)O3)nc2c1 N1(C(C(C2CC2)OC)=O)C2CCCC1CN(C(c1ccc(C)c(F)c1F)=O)C2 CC1CN(C(C2CC(C)N2C(C2CCN2C(C)(C)C)=O)=O)C(C)CO1 N1(C(c2c(OC)ccs2)=O)CC2(CCC(NC(=O)C(C3CCC3)OC)CC2)C1 c1(C(=O)NCC2CC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)ccc(F)cc1[N+](=O)[O-] C1(Cn2cc(CCCC(=O)OC)nn2)CCCCN1C(c1c[nH]c(Br)c1)=O C#CC1(O)CC(C(=O)NCCC2CCCCN2C(=O)Cc2cnnn2C)C1 C(=O)(N=c1cc(Cl)n(C)[nH]1)c1nc(NC(COC)=O)sc1 c1(C(N2CC(NC(c3c(C)[nH]nc3Cl)=O)C(F)CC2)=O)cncc(N=[N+]=[N-])c1 Cc1n[nH]c(=NC2CC3CN(C(c4c(F)ccc(F)c4F)=O)CC23)s1 c1(C(=O)NC2(CC=C)CCN(C(=O)C=CCO)C2)cc(F)c(Cl)c([N+](=O)[O-])c1 C(C(=O)NC(CO)C(C)NC(C1CC(n2ccnn2)C1)=O)(C(C)C)OC C(=O)(C1CNC(=O)c2ccnn21)NC1CC(CCNC(CC(C)(C)O)=O)C1 S(=O)(=O)(c1ccc(Cl)cc1F)NC(CCSC1CC(CC)C1)C(=O)N1CCC1 c1(OC)c(C(N2CCCN(C(C3CC(C)C3)=O)CC2C)=O)ccc2c1CCC2 c1(C(C(N2CC(O)(c3cn(C4CCOCC4)nn3)C2)=O)OC)c(F)cccc1Cl c1(C2C(C(=O)NCC(C)NC(c3csc4cncn34)=O)C2)ccc(F)cc1F c1(C(=O)NC(CC)C)ccnc(CNC(=O)CC2CCCCC2)c1 C(C)(CC(=O)NCC12CC(NC(=O)C(C)Cc3ccccc3)(C1)C2)OC N1(C(c2c(C)nc(CO)o2)=O)CCOCC(F)(CNC(=O)CSC(F)F)C1 c1(CC=O)nc(C2CC2)c(C)s1.CCCCC(=O)N1CC(NC)C1 C(=O)(C(C)(C)CF)N1C(CN(C)C(C2CC2C(C)(F)F)=O)CCC1 Cc1ccc(C(=O)NC23CC(NC(C4CC45CCCOC5)=O)(C2)C3)c(N)c1F c1(C(=O)NC2(C3CN(C(C4(C=C)CCC4)=O)C3)CC2)cccc2ncc(C)n12 c1(C(=O)NC(CN(C(=O)CN2CCCCC2=O)CC)C)cc(C(F)(F)F)cn1C N1(C(c2ncc(CC)nc2)=O)CCCC2CN(C(=O)C3CC3)CCCC12 N1(C(c2c(OC)scc2)=O)C2CCC1CC(C(N1CCCC13CCOC3)=O)C2 Nc1nc(Cl)cc(Cl)c1C(N1CCC(C(F)(F)F)C(NC(=O)CCCF)C1)=O C1(CCCC)CN(C(C=CC(=O)N(C)C)=O)CCN1C(c1c(C)nn(C)c1F)=O C(=O)(CCCCCOC)N1CC(CCNC(=O)CCn2c(C)csc2=O)(OC)C1 C1(C2CN(C(C3CC3c3ccoc3)=O)C2)(NC(C2N(C)CCCC2)=O)CC1 CC1CN(C(=O)CC(C)(C)N2CCOCC2)CCCO1 n1(CCCOC)nnnc1C(c1cncn1C(C)C)NCCS(C)(=O)=O C(CCC(C)C(=O)NCCc1ccc(CNC(=O)C=Cc2ccco2)cc1)OC C1(CC(=O)NCCCF)CC(O)CN1C(=O)Cc1ccccc1 N1(CC)CCN(C(C23CC(CO)(CN2C(=O)C2=C(Cl)CC2)C3)=O)CC1=O C1(NC(COC(CC)(C)C)=O)CCCN(C(c2cn(C(C)C)nn2)=O)C1C CCC(CCC(=O)N1CCC(C(=O)NCc2nncs2)CC1)OC CS(=O)(=O)c1cccc(CN2CCC(F)(C(=O)NCc3ccccn3)C2)c1 CCCC(CCC)C(=O)NC(C)(CNC(=O)CCCN1CCCC1)CC C(=O)(C(CNC(C1CC2(CCO1)CC2)=O)C(C)(C)C)NC(CC=C)CC c1(C(N2CCC(NC(c3c(C)ncn3C)=O)C2)=O)ccc2scc(Br)c2c1 c1(C(N(CC(CNC(CC2C(C)=NNC2=O)=O)O)C)=O)c2ccccc2nn1C c1(C(=O)NCC(C)CNC(=O)CNS(=O)(=O)C2CC2)cc(C#N)c[nH]1 c1(CNC(C23CCCC2(CO)C3)=O)cccc(CNC(=O)C(O)C2CC2)c1 N1(C(CN(S(C)(=O)=O)C)=O)CCC2(CC1)CC2NCc1cccs1.C1(=O)CN1 c1(C(=O)NC(C#C)C2CC2)cccc(-n2cc(-c3cnc(OC(C)=O)s3)nn2)c1 N1(C(c2ccc(OCCC)cc2)=O)CCN(C)C(CNC(=O)C(COC)OC)C1 CCC(C)(C)CC(=O)NCC(C)(CNC(=O)CCC(C)N(C)C)OC Cc1ccccc1COCC(=O)NC1(C)CN(C(C2CCC(C)(CC)O2)=O)C1 c1(C(N(C(CNC(C2(CC(=O)OC)CC2)=O)C)C)=O)oc(NCC2CC2)nc1C c1(CN2C(C(=O)Nc3c(CC(=O)OC)cccc3)CC(O)C2)cccc(F)c1Cl N1(C(c2nc(C)sc2)=O)CCN(C(c2cc3n(c2)CCC3)=O)CC12CC2 C(CC(C)(C)C)(C(=O)N(C)CC1CCCN1C(c1cc2ncccn2n1)=O)OC CC1CCN(C(=O)CCc2cncs2)C(C)C1NC(=O)CCC12CCC(CC1)C2 CC(C)CCCCCC(=O)NCC1CN(C(=O)C=CC(C)(C)C)CC12CC2 C1(NC(C(N2CCC(C(N)C(F)(F)F)C2)=O)=O)COC2(COC2)C1 C12(NC(c3cc(CCOC)on3)=O)CCC(C1)N(C(c1ccc(C)nc1C)=O)C2 c1(N(C(C)CNC(c2cn(C(C)(C)C)nn2)=O)C)cc(C2CCC2)nc(Cl)n1 C1(NC(CN(C(C(C(C)C)SCC)=O)CCOC)=O)CC(C)CC(C)(C)C1 C1(NC(c2coc(C(F)(F)F)n2)=O)CC(O)CN(C(c2cnc(Cl)s2)=O)C1 N1(C(c2sc(Br)cc2Cl)C(=O)NCCC#N)CCN2CCC1C2 C1(OCCC)CCC(N=c2nc3sccc3c(N(C)CC3CCCO3)[nH]2)CC1 C1(OC)CN(C(=O)CC2CC2)CC1C(=O)NC1(c2cncnc2)CC1 C1(C(=O)N=CCCC(=O)N(CCC)CC2CC2)OC2CCC1C2 c1(C(C)CC(=O)N(CCCCNC(=O)C(C)(C)c2cccs2)C)ccccc1F CN1CCC(NC(=O)OC(C)(C)C)(CNS(=O)(=O)CCC2CCCO2)C1 c1(C(N(C)CCN2CCC(S(=O)(=O)N(C)C)CC2)=O)cccc2c1OCCO2 c1(CNC(=O)Nc2cncc(OC)n2)ccnc2c1CCCC2 c1(CC(N2C(CCCNC(c3n(CC)ccc3)=O)CCC2)=O)ccccc1Cl C(=O)(C1=C(Cl)CCOC1)NCCC(C)CCNC(=O)CNC(c1cccs1)=O c1(OCCOC)ccc(-c2nc(C3CCC(F)C3)n(C(C)COC)n2)cc1 c1(OC)cc(C(N2CCCC2CCC(=O)Nc2cnc(Br)c(C)n2)=O)cc(C)c1 CC(C)CC(C(=O)N(C1CN(C(c2nccc(C(N)=O)n2)=O)C1)C)n1ccnc1 Nc1ccc(Cl)c(C(=O)NC2CC(O)CN(C(=O)CSC(F)F)C2)c1 C1(COCC(=O)N(C2CCN(C(C3(C(C)(F)F)CC3)=O)C2)CC)CCCN(C)C1 N1(C(c2ccc(COC)[nH]2)=O)CCC2(CC1)CN(C(=O)C(C)(C)C1CCCC1)C2 c1(OC)cccc(NC(=O)C(C)(C)OC)c1.C(CC)OCCNC(=O)COC c1(C(N2C3C(C(=O)NC4(c5cccs5)CC4)C(C3)C2)=O)ccn2cncc2c1 CC(C)C(C)(O)C(=O)NC1CC(C)(NC(=O)COc2ccc(Cl)c(F)c2)C1 C1(NC(CCOCCOC)=O)CN(C(=O)CC(O)CC2CC2)CC1C c1(C(N(C(c2coc3c2CSC3)=O)Cc2c(C)ncs2)=O)cnc2ccccc2n1 c1(C(N2CC=C(CNC(CC3C(OC)CC3)=O)CC2)=O)nccc2cccnc12 N1(C(CC)CC)CC(C(N2CCC(NC(C3NC(=O)OC3C)=O)CC2)=O)CC1=O C(C(C)(C)C(=O)N1CC(F)(C(=O)N(C)CC2CCOC2C)C1)NC(C)=O c1(CCC)cccc(C(=O)NCCCN(C)CCN(CC)CC)c1 Cc1cc(C(=O)NC2(CF)CN(C(c3cc4n(n3)CCCC4)=O)C2)c(N)c(C)c1 c1(-c2cn(C(C(=O)NCc3c(OC)cccc3F)C)nn2)ccc2c(c1)CCN2 C1(C(N(CC)CC)=O)CCCC1NC(C1CCCN1CC)=O C1(NC(C2(C(C)(C)OC)CC2)=O)CC2CCC1N(C(C1CCCC1(F)F)=O)C2 Cc1cccnc1CC(N1CCCC1(C)C(=O)NCCCC1CCOCC1)=O C12(CNC(CN(C(=O)OC)C)=O)CC1CN(C(c1cc(C)c(C)s1)=O)C2 c1(NC(C)C)cccc(C(=O)NC2(CNC(C3CCCOCC3)=O)CCOC2)c1 C(=O)(C(CCC1CC1)N(CC(C)(C)OC)Cc1ncccn1)OC C1(CNC(C=C(CC)C)=O)CN(C(C2CCC3CC2C3(C)C)=O)CC2(CCC2)O1 CC1=C(C(=O)NC(C)CCN(C(=O)C(O)CCc2ccccc2)C)CCCC1 n1(CC(=O)NCC(C2CCCCC2)NC(CCC=CC)=O)cnc2c1CCCC2 C1(CNC(CC=CCC)=O)(NC(c2ccnnc2C)=O)CCCCC1C c1(C(=O)OC)cc(C(=O)NCC23CC(NC(=O)C(F)C(F)(F)F)(C2)C3)c(F)cn1 c1(C(N2CC(CNC(C(C)C#N)=O)C(C)(C)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 CC(CC(=O)N1C2CCC(C2)C1CC(N1CC(=O)NC(CO)C1)=O)C(F)(F)F N1(C(C=CCC)=O)CCC2CCN(c3nc4ccc(OC)cc4s3)CC2C1 C1(CNC(C(C)C)=O)CN(C(c2c(O)ccc(F)c2Br)=O)CCC1(F)F O=C(C1=NOC2COCC12)NC(c1cccnc1)C(=O)NCCCC1CCC1 CCCCCCC(CC)C(=O)NC(C1CCCCC1)CNC(=O)CCC1CC1 C=CC(C(=O)NCC1(F)CN(C(C2CC2C(C)(C)O)=O)C1)OC c1(CC(=O)NCC(N(C(CCCSC)=O)C)C2CC2)csc2nccn12 C(CCC(=O)NC1(CCCNC(=O)C(C)(C)N(C)C)CC1)OC(C)=O C1(COC)CC2(CCC2O)C1.c12ccc(cc1)CNC(=O)CN(CC)C2.OC c1(C(N2CC(C)C(CNC(c3nncs3)=O)CC2)=O)cc(Cl)cc(Cl)c1F c1(OC)ccc(C(=O)NCCOCCNC(c2cn(C3CC3)nn2)=O)c(CO)c1 c1(CC)cccc(CNC2CN(C(=O)Nc3ccc(CC)cc3)C2)c1 C(=O)(C(C)(C(F)F)c1ccccc1)NCC(CNC(COCC(=O)NC)=O)(C)O N1(c2ncc(COC)cn2)CC2(CCC2)CC1CNC(=O)C=C(C)c1cccs1 CCC(CC)C(=O)N1CCOCC1C(=O)NCCCn1ccnn1 C1(C(N(C(C)C(=O)NC(C)C#C)CC#C)=O)CC(=O)NC1=O N1(C(C2C(CC)CCN2C(c2cnccn2)=O)=O)CCCC2(CCCO2)C1 C1(C(=O)NCCN(C(C2CCCS2)=O)C2CC2)CCc2ccccc2CC1 N1(Cc2ccc(C)cc2C(F)(F)F)CC2CC1(CO)CN2C N1(C(c2cc[nH]c2)=O)CC2CCN(C(c3cccc(Br)c3F)=O)C2C1 N1(C(c2c(OC)cccn2)=O)CC(C(=O)Nc2cc(C)cc(Br)c2)CC(F)C1 CC1C(NC(c2cc3occc3s2)=O)CCCN1C(=O)CCCCNC(N)=O C1(C(=O)NCC2(C)CCCCC2)CC2C=CC1N(C(=O)Cn1cc(C#N)cn1)C2 c1(C(N(C)CC2CN(C(COC(CC)(C)C)=O)C2)=O)cc2c(C)cc(C)nc2s1 CC1(C)C(NC(N2CCC(OC(C)(C)C)CC2)=O)CC1CNC.c1(O)ncccc1F Cc1cc(NC(=O)C(Cn2cccn2)NC(=O)CCCCCF)cc(C)c1C c1(C(=O)OC)nn(C)cc1C(=O)NC1CCN(C(=O)CCOc2cccnc2)C1 CCCC(CNC(c1cnn(CCF)c1)=O)NC(=O)CCC1CC1C c1(C(=O)NCC2CCN(C(C3C4CC5C(C4=O)C35)=O)C2)cn2ccsc2n1 C1(C(N2CCC(CNC(C3CCCN3C)=O)C2)=O)(OC)CCCOC1 C1(CC(=O)NCCn2ccc(C(=O)NCC(C(C)C)C)c2)CC2CCC1O2 C1(C(N2CC=CC(NC(c3cc(OC)no3)=O)C2)=O)CCCC(F)(F)C1 c1(C(N2CCC(CC)(NC(C3CC3F)=O)CC2)=O)ccc2c(c1)CCCS2(=O)=O C(C(C)(C)C#CC(=O)NC12CC=CC(C1)OC2)NC(c1cc(CC)ncn1)=O C1(CNC(C(=O)NCC)=O)COCCN(C(c2cc(C#N)oc2C)=O)C1 c1(CNC(C2N(C(C(CC=CC)CC)=O)CC2)=O)ccnc(P(C)(C)=O)c1 c1(C(=O)NC2CC(NC(CN(C)C)=O)C23CCC3)nn(C)c2ccc(F)cc12 c1(NC(C(=O)NCCSC2CC(O)C(O)C2)=O)c(F)cccc1Cl C1(c2n(C)ccn2)CN(C(C2(C)CC=CCO2)=O)CC1NC(c1cccnc1)=O C(CSC)(CN=c1cc[nH]cc1S(=O)(=O)N(C)CC1CC(C)(C)CO1)OC CCCS(=O)(=O)C(C)C(=O)N(C1CN(C(=O)CN2CCN(S(C)(=O)=O)CC2)C1)C Cc1cnn(C)c1C(=O)NC1CC2(C1)CC2NC(c1ccc(F)s1)=O C1(C(N2CCC(CC(C)O)CC2)=O)C2CC3C(C2NC(=O)CC2CC2)C13 C#CCC(CC#C)C(=O)NC12CC1CN(C(c1cn(CCC(C)(C)C)nn1)=O)C2 CN1CCC(C)(C(=O)NCC2CCCN2C(c2cc(C(N)=O)[nH]n2)=O)C1 c1(NC(c2ccc(CCC(=O)Nc3ccc(F)c(O)c3)[nH]2)=O)ccc(F)c(F)c1Cl CC1OCC2(CCC(CNC(N3CCCC3c3ccc(Cl)s3)=O)O2)C1C c1(C(C)=O)ccc(NC(=O)CCCn2ccnn2)cc1C#N C1(C2CC2)(CNC(C(CC)OC)=O)CCN(C(c2ccc[n+]([O-])c2)=O)C1 C1(NC(c2cnc(C(=O)OC)s2)=O)CCCC(NC(C2CC(=O)NC(=O)C2)=O)CC1 c1(NC(=O)NC(C)C)ccc(C(=O)NC(C)CNC(=O)C(C)C(C)O)cc1 C1(NC(C(CC)NC(C)=O)=O)C2CC1CN(C(=O)C=CSCc1ccco1)C2 CCC(C)C(C)C(=O)NCCC1(NC(=O)CSCCN(C)C)CCC1 c1(OC)ccccc1C=CC(=O)NC(C)(CNC(=O)C=C(C)C)C1CC1 N(C(=NC1CCC1)N1CCOCC2(C1)CC2(F)F)C1CCC(CC(=O)OC)C1 C1(C)(CC)CC(NC(=O)CC(=O)NC)CN1C(=O)CCNS(=O)(=O)c1cccs1 Cc1cc(F)c(N)cc1C(N1CCCC(NC(c2nccc(Cl)c2C)=O)CC1)=O N1(C(c2c(C)cnnc2)=O)CCC(C)(C)C(NC(C2CC(C)(C(C)(C)C)C2)=O)C1 CC(C(=O)NC1CCCC(C(N2CC(C)(C)C2)=O)CC1)S(C)(=O)=O C(=O)(C1=CCN(C(c2cccc(C)c2C)=O)CC1)NC(C#CCCC)(C)C CCC(C(=O)N1CCC(Oc2ccccc2)C1)N(C)C(c1ccn(C2CC2)n1)=O c1(C(=O)NCC(CNC(COCCCOC)=O)F)cn(CC(F)F)nc1C CCCC(C)(O)C(=O)N(CC(O)CN(C)C(c1ccc(NC(C)=O)cc1Cl)=O)C CCCCC(C)(F)C(=O)NC1CC(NC(c2cc(O)nc(N(C)C)n2)=O)C(O)C1 N1(C(c2c(OC)cc(Cl)cc2)=O)CCN(C(=O)C(C)n2cncn2)CC(C)(C)C1 C1(CC(=O)NCC2CCCN2c2nnc(C(F)F)o2)CCC=CCC1 C(=O)(N(CCO)OC)C1(C)N(C(C(C)OCC#C)=O)CC=C1 C1(C(=O)NCC(C2CC2)NC(CSCCC)=O)CCC1(C)C c1(OC)cc(C(N2C(C)C3CC2C3NC(C2CCOCC2)=O)=O)ccc1C c1(C(=O)NCC(CNC(C(COc2ccccc2)OC)=O)O)ncc(C)cn1 Cc1cnn(CCC(N2CC(CO)(NC(C3CC3C#N)=O)C2)=O)c1 c1(N2CCC(C(=O)NC(CCCC(C)C)C)CC2)ncc2c(n1)CCCC2 N1(C(c2c(CC)ncs2)=O)CC(NC(c2ncc(C)cc2OC)=O)C(N=[N+]=[N-])C1 c1(CNc2c(C(=O)Nc3ccc(C)nc3CO)scc2)c(Br)ccc(Cl)c1F C1(CNC(CNS(CC)(=O)=O)=O)CCC2(CN(C(c3cncc(CO)c3)=O)C2)O1 c1(CS(C)(=O)=O)cccc(N(c2nccn2Cc2ccccc2)Cc2cnn[nH]2)c1 C1(CNC(C(C(C)C)OC)=O)CCCC2CN(C(c3ccc(O)cc3F)=O)CC12 c1(C(=O)NCC2N(C(C(CC=CC)C)=O)CCC2)coc2cccc(O)c12 CC(C)(C)CC(O)C(=O)N1CC(C2(Cc3nnnn3CCC(F)(F)C(F)F)CC2)C1 C1(NC(Cc2nc(C(C)OC)sc2)=O)CC(O)CN(C(=O)CN2CC3CC3C2)C1 C1(CCC)CN(C(=O)CCCc2ccccn2)CCN1C(C1CC(C(F)F)C1)=O N1(S(c2cnc(C)n2C)(=O)=O)CCC2(O)CCCCC2(O)C1 c1(NC(=O)CC2(NC(=O)Cc3cccc(O)c3O)CCC2)cccc(Cl)c1Br N1(N(CCC=C)C)CC(F)(F)C(F)(F)C1 c1(CC)nc(=N)[nH]c(=NC(CNC(=O)Cc2ccc(CO)cc2)C(F)(F)F)[nH]1 CCCC(CCC)CC(=O)NCC1CCCC(CNC(C2CC(C)CCO2)=O)C1 c1(C(=O)NCCN(C(c2noc(CC)c2C)=O)CC)c(C)cc(OC)cc1F C(=O)(C(F)(F)C(O)C1CC1)N1CCN(C(CNC(c2cn(C)nc2Cl)=O)=O)CC1 c1(CC)oc(C)cc1C(N1CCCC1CN(C(=O)CC(=C)C)C)=O c1(SCCC(=O)N(C)CC2CN(C(c3coc(CO)c3)=O)C2)ccc(Cl)cc1 N1(C(c2c(C#C)cn(C)n2)=O)CC2CCC1CN2C(=O)CC1CCOC1(C)C C(C(C(=O)NCC(C)CNC(C1(C(C)C)CCC1)=O)C(F)(F)F)OC N1(C(C(C)SCCCC)=O)CCCC(CN(C(=O)Cn2ccccc2=O)CC)CC1 c1(CC)c(C(=O)NCCCCNC(=O)C(C)(C)C)cnn1-c1cccc(C)c1 N1(C(c2c(C)sc(Cl)n2)=O)Cc2ccc(CNC(=O)CC3CCC(O)C3)cc2C1 C1(OC)CC2CC(NC(C3(C(N)=O)CC3)=O)C1C2.C(=O)(C(C)(C)n1ccc(SC)n1)N C(Cn1ccnc1)(CN=c1[nH]c2c(c(=NCc3cnc[nH]3)[nH]1)CSC2)OC N1(C(C(CC)O)=O)CC(C(=O)N(CCn2ccnc2)CC)C2(CC2)C1 C(=O)(C(=O)C(C)(C)C)NC1CN(C2CN(C(CS(CC)=O)=O)C2)C(=O)C1 N1(C(C2CCC=CO2)C(=O)NCC2CCCCC2)CCC12CCCC2 Cc1cc(C(N2CC(N(C)C(c3ccsc3C#N)=O)C(F)C2)=O)cc(Cl)c1 C12(C(=O)O)CCC(C(=O)Nc3cc(CN4CCCC45CC5)c(F)cn3)(CC1)CC2 c1(C(N2CC3C(NC(C(C)NC(CC)(C)C)=O)C3C2)=O)cc(C)cc(Cl)c1 CC1CN(C(c2ccc(N)c(Cl)c2)=O)CCC1CNC(C1CCCC1O)=O C(CCCC(=O)NC1CN(C2CC2)C1)n1cc(-c2c(OC)ccnc2)nn1 Cc1ccc(C23COC(C2)C3C(=O)NNC(N)=O)cc1 C1(C)(CC(=O)N(CC(=O)N(C)Cc2cnns2)CC2CC2)CCOC1 c12cnc3c(cccn13)NC(=O)c1sccc1-2.c1(OC)nccc(OC)c1Br c1(COC)nc(NC(C2CN(C(=O)Cc3cnoc3)C2)C)cc(O)n1 CC1(C)CCCCC1C(=O)NCCNC(c1ccc(-c2cccc(Cl)c2)s1)=O c1(C(=O)NC2(C)CC(NC(C(CC)n3ccnc3)=O)C2)cnc2sccn12 N1(C(CC(C(C)C)O)=O)CC(C(=O)NCC(O)COC(C)C)C2(CCC2)C1 C12CCCC(C1)N2.Cn1nncc1CNC(C12CC(NC(=O)CNC=O)(C1)C2)=O C12(NC(C3(CC)CCCCC3)=O)CCCC1N(C(c1cc(C)c(Cl)s1)=O)CC2 c1(C(N(CCNC(=O)CC2CC3(CC3)CO2)CC)=O)cnn2c1NCCC2 C(=O)(C#CC1CCCCC1)N1CC(F)(CNC(c2c(C)nn(C)c2N)=O)C1 N1(C(C=CC)=O)CCOC2CCN(C(=O)COC3CCCCC3)CC12 C(=O)(C1OCCc2ccccc21)N(C)CC1CCN(C(c2nc(C)oc2)=O)C1 c1(N(CCCCC=O)C)nc2ccc([N+](=O)[O-])cc2s1.C(CCN)SC S(=O)(=O)(c1ccc(NC2COCC2N2CCOCC2)nc1)N1CC(C)(C)C(CO)C1 C(=O)(CC(C)CC(=O)NCCCC(O)C(=O)N1CCOC(C#N)C1)OC O=C1NCc2c(COCc3cn(CC45CCCC4C5(F)F)nn3)cccc21 Cc1nnc(CN(CCCNC(=O)CN2CCCC2CO)C(C)C)o1 c1(C(=O)NCC(=O)NCC2C(CNC(C(C)C3CCCC3)=O)C2)ccccc1 c1(C(=O)NCC2CCC(C)(C)CN2C(=O)C2=CCC2)cc(S(N)(=O)=O)ccc1F O=C1C2CC3C1C3C2C(N1CC=CCC1C(N1CCCC(CC2CC2)C1)=O)=O C=CCC(CC)C(=O)NCC1CN(CC(c2ccc(C3CC3)cn2)=O)CC(C)O1 c1(C(N(C2CCCN(C(c3ccc(C4CC4)s3)=O)C2)C)=O)cnn(C)c1N C1(C(=O)Nc2ncc(C3CCC(C)O3)s2)CCCCCCC1C(=O)O N1(C(c2ccoc2Cl)=O)CCC(C2CCN(C(C3C4CC4C4CC34)=O)CC2)CC1 c1(C(=O)NCC2(C)CCN(C(C3COCCC3(F)F)=O)C2)scc2c1OCCO2 C1(NC(C2CC(O)C2)=O)CCC2(CCCN(C(c3csnn3)=O)C2)C1 c1(CN(CC(=O)NCC(=O)N(C(C)CCC)OCC)C)ccccc1 N1(C(C2C(C)=CCS2)=O)CCCC1(C)CNC(c1ccccc1C)=O C1(C(N2CCC(C(CNC(C3C(C)C3C)=O)(C)C)CC2)=O)C(C)(C)OC1(C)C CCC1=C(C(=O)NCCCCNC(C2CCc3cnn(C)c3C2)=O)SCCO1 C(c1ccsc1Br)=CC(=O)N(C(C)CNC(C1(c2nc[nH]n2)CC1)=O)CC c1(C(c2n(C)nnn2)NC2CCCN(Cc3ccccc3)C2)cc2ccncc2s1 n1(CC=C)cc(C(=O)NC(CNC(c2csc(C(C)(C)C)n2)=O)CC)nn1 C(=O)(C(F)C(C)CNC(C1(C)CCCCC1C)=O)Nc1cc(OC)ncc1 CON(CCC(=O)N(C1CCOC1)C)C(=O)CCOC1CCOC1 C1(c2ccccc2)(NC(COCC(=O)OC)=O)CCN(C(=O)C(C)C2CCC2)C1 c1(CC(N2CC(NC(c3c(CC)noc3C)=O)C(F)C2)=O)coc2ccccc12 c1(C(=O)NC(CC=C)CNC(C2C=CCC2)=O)ccccc1SC(F)(F)F C1(C)(C(=O)NCC2C(C)C2(F)F)CN(C(=O)CCC2CCOC2)C(C)(C)C1 S(=O)(=O)(c1ccc(Br)c(Cl)c1Cl)NC(=NC)NCc1ccccc1N Cc1cncc(C)c1C(=O)NC1CCCN(C(C2(C)COC2)=O)C1 C1(CNC(C(C)=CC)=O)COC(C)(C)CN1C(=O)C(CCC)N(C)C C1(NC(C2CCCC(C)O2)=O)CN(C(=O)OC(C)(C)C)CC1S(C)(=O)=O CC1CC(CCNC(c2cnccn2)=O)CCN1C(C1CN(c2nncs2)C1)=O C1(NC(c2ccc(NC(C)=O)cc2Cl)=O)CN(C(C2(C)CC2)=O)CC1C1CC1 c1(C(N2CCC(O)(C(=O)OC)C2)=O)cc2cccn2cn1 C#Cc1cnn(CC(=O)OC(c2ccc(C(C)C)cc2)(C)C=O)c1.C1C(C)(O)O1 c1(C(N2CC(C)(CNC(C3C(CCOC)C3)=O)C(C)C2)=O)nccc2occc12 n1(CC=C)cc(CCCC(N2CCCC2C2(O)CC2)=O)nn1.CC(C)CO C1(C(N(CCO)CC)=O)CCCC(NC(c2cncn2C)=O)CC1 C(=O)(C#Cc1ccccc1)N1CCC(F)(C(=O)NCCCOC)C1 c1(C(N)=O)ccc(C(=O)NCC2CC2NC(=O)CCF)nc1 C#Cc1cn(C)nc1C(=O)NC(Cc1cn(C2(OC)CCC2)nn1)C(=O)NC Cn1ncc2c1CN(C(C1CCCC1NC(c1cc(Cl)cc(Cl)c1O)=O)=O)CC2 C1(CNC(C(C)CCO)=O)COCCN(C(C2CCOC2)=O)C1 N1(C(C(COCC)C)=O)CC2CS(=O)(=O)CC2(NC(c2ccn(C)c2)=O)C1 C1(N(S(CC=C)(=O)=O)C(C)C)CCC(NCc2ccc(O)nc2)OC1 N1(C(C2N(C(CCC(=O)OCC)=O)CCC2O)=O)Cc2cccc(Br)c2C1 C(CCCCCc1nc(C2CC2(C)C)nn1-c1nc(C)nn1C)OC N1(C(C2CCC(CNC(C3CC(N(C)C)C3)=O)O2)=O)CCc2nocc2C1 C1(NC(C(c2ccccc2)OCC)=O)CN(C(=O)C(Cl)=CCl)C2CC12 c1(CC)cc(C(=O)NCCC2CCC(NC(c3ccsc3C)=O)C2)sc1C C1(CCN(C(C23OCC(COC)(C2)C3)=O)C)Cc2ccccc2O1 c1(NS(CCC)(=O)=O)ccc(NC(=O)Cc2csc(C)n2)c(C)c1 c1(C(=O)NC(C)CC2CCCO2)n[nH]c2c1CN(C(=O)C(CN(C)C)N(C)C)C2 N1(C(C(=O)NCc2cccc(F)c2I)=O)CCC2(O)CCOCC2C1 N1(C(C2(CC)COC2)=O)CC2CCC1CN2C(c1c(Cl)cncc1Cl)=O Cc1nc(O)nc(O)c1CC(N1CCC2CCC12CNC(c1coc(Cl)n1)=O)=O N#Cc1cc(Cl)c(C(N2CCOC(CNC(C3CC3C(F)(F)F)=O)C2)=O)s1 C1(C(N2CCOC(CCF)C2)=O)(CNC(=O)C=CCO)CC12CCC2 c1(-n2c(C(C(CSC)C)(C)NCC(C)(C)F)nnn2)ccc2c(c1)OCO2 C1(N(C(c2cnn(CC)c2C)=O)C)CN(C(c2cncc(O)c2)=O)CCC1C Cc1cc2c[nH]nc2cc1C(N1CCN(C(=O)CCCC2CC2)C(C2CC2)C1)=O c1(NC(=O)CC2CCCC2C(N2CC(c3ncc[nH]3)C2)=O)cccc(F)c1 C1(C(=O)NCC2(NC(C(C)N(C(C)=O)C)=O)CCC2)Cc2nnc(C)n2C1 c1(C(N(CCNC(CCC=C)=O)CC2CC2)=O)ccc(Br)cc1OC(F)F C1(C)(C(=O)NC(CCOC(C)C)C(=O)NC2CCCC(CO)C2)CCC(=O)CC1 C=CCC(C)(C)CC(=O)N1CC(NC(=O)C(=O)Nc2ccccc2)CC1COC c1(C(=O)NC2C(NC(c3c(C(C)C)ccc(C)c3)=O)C2)ccc(Cl)c(F)c1F C(C)(CNC(c1ccn(C)n1)=O)(CC(C)C)NC(C1CC(=C)C1)=O C1(C(N(C2CCCC2)CCNC(C2CC(=C3CC3)C2)=O)=O)CC(F)(CF)C1 N1(C(C2(OC)CC2)=O)CCC(O)(C(C)NC(C2(F)CCCN(C)C2)=O)CC1 CCCCCCC(C)CC(=O)NCC1CCN(C(=O)CCC(=O)NC2CC2)C1 c1(CC(C)Sc2nnc(SCC=C)n2-c2ccccc2)cc2ccccc2o1 N1(CC)CCN(C(C2(OC)CCN(C(=O)CN3CCCCC3)C2)=O)CC1 C1(NC(=O)CC2CC2)CCC2CN(c3nc4ccccc4o3)CC2C1 C1(NC(C2C=CCC2)=O)CCN(C(c2ncc(Cl)s2)=O)C12CCC2 C12(C(N3CCCC(NC(=O)CCC4CCCO4)C3)=O)CC1CCC2(F)F C1(C)(CC)CC(NC(c2cncs2)=O)CN1C(=O)CCc1cn(C)nc1C c1(C(=O)NCCC2CCN(C(C(C)=C3CC3)=O)CC2)cc(F)c(Cl)cc1Cl c1(C(=O)NC2(C)CC(NC(C3CCN4CCCC4C3)=O)C2)cc2ncccc2[nH]1 c1(CN2CCC(C)(NC(C(C)CSc3ccccc3)=O)C2)c(Cl)cccc1C#N C1(CC)(NC(C2CC(CC3CC3)C2)=O)CN(C(C2CCNC2=O)=O)C1 Cc1cn2cc(C(=O)NCC(C(C)(C)C)NC(c3cc(N)cc(F)c3)=O)sc2n1 c1(C2N3CCC(CC3)NC2=O)c(F)cccc1F.CN1CCNCC1 N1(C(CCOCCCNC(c2c(CC)cno2)=O)=O)CCC2OCCC2C1 CCC(C)(C)C(=O)C(=O)N1CCC(C(N2CCC(c3cnn[nH]3)C2)=O)CC1C c1(N(C(C(Cc2cc[nH]n2)NC(c2n(CC)ccc2)=O)=O)C2CC2)ccccc1C N1(C(C)=O)CCN(C(C2C3CN(C(c4cncnc4Br)=O)CC23)=O)CC1 C1(CNC(C(C(C)C)NC(=O)OC)=O)CCN(C(C2(CN(C)C)CC2)=O)C(C)C1 CCCC(C(O)C(=O)NC1CCOC1C)NC(C12COCC1C2)=O c1(C(=O)NC(C)C(=O)N2CC(NC(=O)CC3CC3)C2)cc(OCCO)ccc1Cl C1(NC(COCCC=C)=O)CN(C(c2cc(Br)sn2)=O)CC12CC2 c1(CN(CCOC)Cc2ccccc2)cc(-c2ccc(C)cc2)ccc1F C1(C(C(=O)NCCCN(C(=O)CC(C)(C)C)C(C)C)C)CC2(CCC2)CO1 CCN=C(NCCCCC#N)NCC1(CS(C)(=O)=O)CCOCC1 C1(NC(C(CC)N(C(c2nc(CCC)oc2)=O)C)=O)CC=C(C)CC1 c1(CNC(c2n(CC#C)ccc2)=O)ccc(C(=O)NC2CCCC2SCC)nc1 C1(O)(CNC(=O)CSC2CC2CNC(=O)CC2CCOCC2)CC2CCC1O2 C12(NC(CCNC(=O)OCC)=O)CC(C(=O)NOCC(C)(C)O)(C1)C2 C(=O)(CCC(C)(C)C(=O)Oc1ccccc1)NC12CC(C)(OCC1)C2F N1(C(c2c(C)oc(C#N)c2)=O)C2CCCC1CC(NC(=O)CCOC1CCC1)C2 C1(C(N2CCC(COC)C2)=O)CC(=O)CN1C(C1CC(CC2CC2)C1)=O c1(C(=O)NCC2C(NC(Cc3c(C)occ3)=O)CCC2)cc2c(C)cccn2c1 C1(OC)CC(CCN(C)C)N(C(c2ccc(C3CNC(=O)C3)cc2)=O)C1 N1(C(C2(OC)CCCC2)=O)CCC(C(=O)NC2CC(N3CCCC3)C2)C(C)C1 Cc1nc(Br)oc1C(=O)NC1CC(NC(=O)CCC(=O)c2ccc[nH]2)C1 N1(C(c2cnc(OC)nc2)=O)CC(NC(c2cc(CO)oc2C)=O)C2CCCC12 C12(NC(C(=O)NCC)=O)CCC(C1)N(C(=O)CCc1cccs1)C2 CCC(C)C(CNC(C1(CNC(=O)CC2CC3CCC2O3)CCCC1)=O)CO c1(CC(N2CCN(CCOCc3ccccc3)CC2)C)cccc(Cl)c1 N1(C(C(C)CC#N)=O)CCOC(C)(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 C1(NC(=O)CCn2cccc2)CCC(CCNC(=O)C(O)CN2CCOCC2)C1 N1(C(C2SCCCS2)C)CC(CNC(=O)CCC(C)(F)F)C(C)(C)C1 C(=O)(C(C)(O)CC(F)F)NC(CC=C)CNC(=O)COc1ccc(F)cc1 Cc1cc(OCC(=O)NCCCC(C)NC(=O)CCCCN(C)C)cc(C)c1 c1(C(=O)NCCC2CC(NC(C3OCC(C)(C)C3)=O)C2)ccc(N)cc1O N1(C(c2ccc(CC)s2)=O)CCC(F)(C(=O)N(c2cccc(F)c2)CC)C1 c1(C(N2CC(NC(C3CC34CCSCC4)=O)C(F)C2)=O)cccc2c1OCCN2 C1(C(=O)NC2CC(OCC(=O)NCC3CCCO3)C2)CC(=O)CS1 c1(CC)ccc(N)c(C(=O)NC(CO)C(C)NC(=O)CCn2ccnn2)c1 CCC(C)(C)C(O)C(=O)N1CCC(N(C)C(c2cnc(C)c(N)c2)=O)C1 C1(NC(C)=O)CN(C(=O)C(C)(C2CCOC2)NC(=O)OC(C)(C)C)CC12CC2 N1(C(c2scc(CC)c2)=O)CC(OC)CC1(C)CNC(=O)CN(C(=O)C(C)C)C.CC CC(CC(=O)N1CCC(CNC(C2CC3C=CC2O3)=O)C1(C)C)C(F)(F)F c1(NC(C(C2(C)CC2)NC(C(CC)NC(N)=O)=O)=O)c(C)cc(C)nc1C N1(C(c2c(OC)csc2)=O)CCC2CC2(C(=O)N(C)CC2(CO)CC2)CC1 c1(C(C(=O)NC(CCN(C(CCc2cc(C)no2)=O)C)C)C)ccc(F)cc1F CCC(C)C(CC(=O)NC1CCSCC1)NC(=O)CN(C)C(N)=O C1(NC(c2c(CC)con2)=O)CCC2(CCCN(C(=O)Cc3csc(C)n3)C2)C1 N1(C(CCCC(C)(F)F)=O)CCCC2(CCC(NC(c3ncc(F)cn3)=O)C2)C1 N1(C(c2sc(C)c(C)c2C)=O)CC2(CCCC(CNC(c3ccns3)=O)O2)C1 c1(OC)cc(N2CCC(C)C2CNC(c2cnc(C)s2)=O)nc(OC)n1 C1(C(=O)NCC(C)(CO)NC(c2cc(C)c(O)nc2)=O)CCn2ccnc2C1 C1(CNC(C(C2CCCC2)OC)=O)CCCN1C(c1cnc(-c2nc[nH]n2)s1)=O c1(OC)cnc(F)cc1C(=O)NCC(C)NC(=O)CC1CN(C)CC1O CC1CC=C(C(=O)NC(CC(=O)NCc2cnncc2O)C(F)F)CC1 Cc1cc(O)nc(C)c1C(N1CC2C(NC(=O)CC(C)NC(N)=O)C2C1)=O C1(C(=O)NCCCN(C2CCCC2)C(C2C(C(C)C)C2)=O)CCS(=O)(=O)N1 CC1=C(C(=O)NC(C)(C)CC(F)C(=O)NCC2(C)CCCCCC2)CCCO1 N1(C(C(CC=C)(C)C)=O)CCC(C2CC(NC(c3cc(OC)ns3)=O)C2)C1 Cc1cnn(C(C)C)c1C(=O)NC1CC(NC(C2COC(C)C2)=O)C(O)C1 c1(C(C)OC)nc(C)c(C(=O)NC2COCC2NC(c2cnccc2Cl)=O)s1 C(=O)(C1COc2ccc(Br)cc21)N(C1CCN(C(CC=C)=O)C1)CCO n1(CC)ncc(Cl)c1C(=O)NC1CCOC(CNC(c2sccc2COC)=O)C1 CCCC1=C(C(=O)OCC)C(c2nc(C)ncc2F)NC(=O)N1C(CC)CC CCCC(C(=O)N(C1CCN(C(c2ccc(C(F)F)cn2)=O)CC1)C)OC C1(C(N(C)CC2(NC(=O)CCCC#N)CCC2)=O)CCCC(C)(C)C1 c12cc(cc(Cl)c1OC)C(=O)O2.C(=O)(CCCOC)N(CCN(CCC)C)C c1(CN(C(C(=O)NCC)C2CCSC2)C)ccc(CCC(C)C)cc1 CC(O)(CC(=O)N1CCCC(O)(CNC(=O)CCc2ccncc2)C1)C(F)(F)F c1(C(N2CCC(N(C(C(=O)NCCOC)C)CC)CC2)=O)cc2ncccc2o1 c1(C(=O)NC2CCC2NC(c2c(F)cccc2Cl)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] c1(OCC)ccccc1C(N1CC2C(NC(c3cnc(SC)s3)=O)C2C1)=O N1(C(C2=CC(C)(C)C2)=O)CCCC2CCN(C(=O)COC(F)F)CC12 C1(NC(C2C(C)CCS2)=O)CCC(NC(c2cnn(C3CCCC3)c2)=O)CC1 Cc1cc(F)cc(C(N2CCC(CNC(c3cc4cccnn4n3)=O)C2)=O)c1C C12(C(N(CCC(N3CCC4CC(CC)C4C3)=O)CC)=O)CC3CC(CC(C3)C1)C2 c1(C(N2CCC(O)(CCNC(c3cc[nH]n3)=O)C2)=O)c[nH]c2cccc(Br)c12 C1(C(=O)NCCC(=O)NCCCC(=O)OC)CCCC(N)C1 C12(C(=O)NC(=O)NCC3C(OCC)C3)CCC(OC)C1C2.C12CC(F)(C1)N2 CC1CC(C)(C)CN1C(CC1(C#N)CCC1)C(=O)NC1CCC1 N1(c2ccc(C(=O)OC)cn2)CCC(C)C(NC(c2ccoc2OC)=O)C1 C(C(C)(C)CC(=O)N1CCCC(CNC(=O)CN2CCCC2C)CC1)OC C1(NC(=O)CCCc2ncco2)CC2CCC1CN2C(=O)CCF C=CC(C)(CCOC)C(=O)N1CCC(CNC(c2cnn(C3CC3)c2Cl)=O)CC1 N1(C(C(CCOC)C)=O)CCCCCC(NC(c2cc(C(F)(F)F)ns2)=O)C1 OC1CCCN(C2CCN(S(=O)(=O)C(F)(F)F)CC2)C1 Cc1ccc(C(C)C(=O)N(CCN(C(C2CN(C(C)C)C2)=O)C(C)C)C2CC2)s1 N1(C(C(C)n2cccc2)=O)CCCC(CNC(c2cc(F)n(C)n2)=O)C1 c1(COC)ccc(C(=O)NCC(O)CN(C)C(c2cc(C)sc2C)=O)cc1F N1(CCNC(C2CCCO2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC12CCC2 C1(NC(=O)Cc2cnns2)C2CCC1N(C(c1cccc(Cl)c1)=O)C2 C1(NC(c2cncc(C)c2)=O)CC2CC1CN(C(C13CCC(CO)(CC1)C3)=O)C2 C1(NC(CNC(=O)OC(C)(C)C)C2CC2)CC2C=CC1C21CC1 C(=O)(CC(O)C(C)(C)C)N(C1CN(C(c2cnccc2Cl)=O)CC1O)C C(C(F)(C(=O)NC(C12CCC(CC1)C2)C)C(C)C)NC(c1cccc(OC)n1)=O C(=O)(C1CCc2ccccc21)N1C(C)(C(=O)NC2CCC(O)C(O)C2)CC(O)C1 c1(OCCN(C(=O)C(F)(F)CSCCO)C)ccc(C(C)(C)C)cn1 Cc1cc(C(N2CC(C(=O)NC3CC(=O)NC3=O)C(C)C2)=O)[nH]c1C c1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(Cl)cn2)ccc2nsnc2c1 CCC(Cc1nc(CCSC)nn1-c1cccc(C(C)C)c1)C(F)F N1(C(c2c(C)cc(N)cc2)=O)CC(NC(C2CCC(C)O2)=O)C(C2CC2)C1 C#CC1CCN(C(=O)CCN(CCO)C(c2cn(CCOC)nc2C)=O)C1 c1(C(N2CC(CCNC(C3CCC4(CC4)C3)=O)OCC2)=O)ccc([N+](=O)[O-])cn1 N1(C(c2c(OCC)scc2)=O)CCc2sc(CNC(=O)C(C)(C)C#N)nc2C1 N12CCC(C1)C2=O.C(C)(C(=O)NC1(CC=C)CCC1)=CC=C C=CCC(C)(C)C(=O)NCC(C)(C)CNC(=O)C=C(C)c1ccsc1 C(=O)(C(O)CC(C)(C)C)NCCC1(C(N(CC#C)CC2CCCO2)=O)CC1 O=[N+]([O-])c1cc(F)c(C2CCCCN2CCO)cc1Br.C12CC13CC2C3 c1(-c2n(CC)nc(C)c2)ccc2c(C(=O)Nc3ccccc3C(N)=O)n[nH]c2c1 c1(NC(CNC(N)=O)=O)cccc2cnccc12.c12cnc(Cl)cc1C(=O)N2 CC(=O)CCC(=O)NC(C)C=CC(N1CCCC1c1ncc[nH]1)=O c1(N(C(CCCC)=O)C)nc(-c2cc(N3CCCC3)ccn2)nn1CC1CC1C C(=O)(CCCCCC#N)N1CCC(CNC(C(Cc2ccccc2)OC)=O)CC1 Cc1cc(C(=O)NC2CCCC(N(C)C(c3cc(O)ncn3)=O)C2)cc(Cl)c1 c1(C(N2CC(NC(CC=C)=O)C(N=[N+]=[N-])C2)=O)ccc(C)c2[nH]c(C)cc12 N1(C(C(C)Cn2cccn2)=O)CCCC1(C)CNC(c1cc(C(F)F)nn1C)=O c1(C(C)F)cccc(NC(=O)C(=O)NCC2CCCOC2c2ccc(C)cc2)c1 Cc1cc(N)c(C(=O)N(C)CC2CCN(C(=O)C(C)C3CCC3)C2)c(F)c1 c1(C(=O)NC(C(C)NC(C(Cc2c(C)nc[nH]2)O)=O)CO)cccc(O)c1Cl c1(C(=O)NC(C(=O)NCCC(CC)(F)F)C(C)CC)ccn2cncc2c1 c1(NC(c2cocn2)=O)cccc(-c2cnc(N3CCCC3)nc2)n1 N1(C(Cc2c(Cl)cn(C)n2)=O)CCC2(CC1)CN(C(=O)C(c1ccccc1)F)C2 c1(C(N(C)CC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)cnn2cnnc2c1 C1(CCC)CN(C(c2cnc(C3CCOC3)s2)=O)CCN1C(=O)Cn1cnnn1 C1(C(=O)NC(C(C)NC(c2cnc(-c3ccncc3)s2)=O)C)(CO)CCOCC1 N1(C(C(C=C)C)=O)CC2CC2(C(=O)NCC2CCOC2(C)C)C1 c12ccccc1CN(C1CC1)C(=O)CO2.C1(C(C)C)CCCO1 N1(C(c2c(C)noc2N)=O)CCC(C(N2CCC(O)(C(C)C)C2)=O)C(O)C1 CN=c1[nH]c(=NCCN2CCCCC2C)[nH]c(=NCC=C(Cl)Cl)[nH]1 C1(CCNC(COCCC#C)=O)CN(C(=O)CCOCCOC)CC(C)O1 C(=O)(CCCCN1CCOCC1)NCC(CC)NC(c1ncccc1OC)=O n1(CCOC)cc(C(=O)NC2CC(CC(=O)NCCCc3nncs3)C2)nn1 c1(OC)cccc(C(C)CC(N2CCC3C(NC(=O)CSCCN(C)C)C23)=O)c1 C1(NC(c2cnn[nH]2)=O)CN(C(=O)CCOc2ccccc2)C2(CCC2)C1 c1(NC(N2CCOC(C3CC3)C2)=O)cccc(CO)n1 N1(C(CC2C(C)C2)=O)CC(C2CCCN(C(=O)C(C)Sc3ccc(F)cc3)C2)C1 CC1CSCCN1C(C1(CNC(=O)C=Cc2ccoc2)CC(C)(C)C1)=O C1(NC(c2c(C)ccnc2)=O)C(C)(C)C(C(=O)NC23COC(CF)(C2)C3)C1(C)C N1(C(C(C)NS(C)(=O)=O)=O)CC2CC(NC(c3cc(Cl)c(Cl)n3C)=O)C1C2 CCCS(=O)(=O)CC(=O)NC1CCC(C)N(CCC2CC2(Cl)Cl)C1 N1(C(C(C)NC(=O)NC)=O)CCN(C(=O)CC2(C)CCOCC2)C(C)C1C c1(CC)ccc(F)cc1C(=O)NCC1CC(O)(CNC(=O)CS(N)(=O)=O)C1 c1(C2CCN(C(CCOC(C(CC#C)C3CC3)=O)=O)CC2)cc2ccccc2o1 c12ccnc(c1)N(C(c1ccccc1)C)C(=O)Cc1cn-2nn1.C(C(=O)O)OC C1(CC)CCN(C(c2cccc(Cl)c2)=O)C1CNC(=O)C(C)NC(C)=O N12CCCCC1CNC(=O)C(C)CNC(=O)C2.c1(CON)ccccc1 CCCCC(CC)CC(=O)N1CCC(C)N(c2nccc3ccsc23)CC1 N1(C(C#CC(C)(C)C)=O)CCC2(CC1)CN(C(C1CCn3ccnc3C1)=O)C2 C(=O)(C1CCc2c[nH]nc21)OCC.C1(=O)C(CC)(CC)OC2(C#N)CN1C2 N1(C(C2(C#N)CCSCC2)=O)C2CCC1C1CC1(NC(C1CC3C=CC1C3)=O)C2 n1(CC)nc(C(N2C(C(=O)Nc3cccc(COC)c3)CC2C)=O)cc1C c1(COCC(=O)NCC(CN(C(C(F)=CC)=O)C)C)ccc(C(F)F)cc1 C1(C(=O)NC(c2cccnc2)CC)CSCCN1C(c1ccnc(C)c1)=O c1(OC)ccc(-c2cccc(CC(=O)OC(N3CC4(CCC4)C3)=O)n2)cc1 C1(CC(=O)NC(CNC(=O)CN2CCCCCC2)C2CC2)CC(F)(F)C1(F)F C(=O)(C(C)(C)CC(C)C)N1CC2CC(CNC(c3c(C)nc(=N)[nH]c3)=O)(C2)C1 c1(OCC(=O)NC2C(NC(CC=CC=C)=O)CCC2)cccc(C)c1F C(=O)(CCCc1ccccn1)NCCC(C)NC(C(C)=C1CC1)=O c1(NC(=O)NCCN(C(=O)COc2ccccc2)C)ccc(C(C)CCO)cc1 C1(O)(CN(C(=O)CSCCC(F)(F)F)C)CCCN(C(=O)CN2CCNC(=O)C2)C1 c1(CN(CCC)C(=O)NC(C2CCCN(C)C2)C)ccccc1Br C#Cc1cc(OC)cc(C(C(=O)NC(C)C)N(C2CCCC2)CC2CCOC2)c1 N1(C(C2(CC)CCC2)=O)CCC(NC(c2ncc(C)cc2F)=O)C(C(C)C)C1 C1(NC(c2n(CC)cnn2)=O)C(C)CCN(C(=O)CC2CCCCO2)C1C N1(Cc2c(OC)ccc(Cl)c2)CCC2C1CCCN2C(c1cc(O)cc(O)c1)=O c1(C(=O)NC(c2cocn2)CC)c(NCc2cnc(OC)nc2)cccc1F N1(C(C2CC3(CCC3)CO2)C(=O)NCC(=C)C)CCc2ccc(C)cc21 n1(CC(=O)NCC2(F)CC(NC(c3ccsc3Br)=O)C2)cnnc1O C1(CNC(C(C)OCC#C)=O)CC(F)(F)CN1C(C1CCOC(C)(C)C1)=O N1(C(CC=C)=O)CCC2CN(Cc3ccc(O)c(C)c3O)CC12 CC(C)CC(C)CC(=O)NCC1CCN1C(=O)C(C(C)O)N(C)C CCCC(C)C(=O)NCCN(C1CCCCCC1)C(c1cnn(CCO)c1C)=O CC(C)C(C)(CNC(C1(C2CC2)CC1)=O)NC(c1cnn(C2CC2)c1)=O Cc1nc(CC2CC2)oc1C(=O)N(CCC(C)(C)NC(=O)C1=NOCC1)C C1(NC(C2C(C)(Br)C2)=O)CC2(CCC(CNC(c3cccc(CO)c3)=O)OC2)C1 N1(C(C2SCCN(Cc3nc(C)oc3)C2)=O)CC2CC2C1C#N C(=O)(CC1=CCN(C)CC1)NC1(CC=C)CN(C(=O)C(O)C(C)(C)CC)C1 C1(N(C(=O)CC2CC2)CCC)CCN(C(=O)C(F)CC2CCC2)C1 c1(N2CC3C(NC(=O)C(O)Cc4cnc[nH]4)C3C2)nccc(C(N)=O)c1[N+](=O)[O-] Cc1cc(C(N)=O)ccc1S(=O)(=O)NC(=O)C=Cc1cccc(C#N)c1 N1(C(C(CC)(C)COC)=O)CC2(CCN(C(=O)CCC3CCOCC3)C2)C1 c1(C(N2CC(C=C)C(NC(=O)C(O)C3CC3)C2)=O)cc(OC)cc2cccnc12 N1(C(CC2N(C(C)C)CCC2)=O)CCCC(c2cn(CC3CCO3)nn2)CC1 C1(C#N)(C(N(CCCCNC(C2CCC2C(C)(C)C)=O)C)=O)CC2CC2C1 N1(C(CCC(=O)NC)=O)CC2CC(C1)CN(C(=O)C(C)c1cncs1)C2 CC(C)C(C)(C)C(=O)NCCOCCN(C(=O)CSc1ccc(Cl)cc1)C c1(C(C(=O)NCC2CCC(O)CC2)NC(C(COC)(C)C)=O)c(C)cccc1C C1(C(N2C(C(=O)NC3C=CC(CO)C3)CCCC2)=O)CCC2CC1CO2 C1(NC(CCC)=O)COC2(CNC(C3CCCN3C(c3ccco3)=O)=O)CC1C2 N1(C(=O)CSCc2ccccc2F)CC2(C1)CN(C(N1CCCC1)=O)CCO2 C12(C(=O)NC3(CSC)CC3)CC1CN(C(=O)CC(C1CC1)OCC)C2 N1(C(c2c(C)nco2)=O)CCN2CCN(C(C3CCCSC3C)=O)CC2C1 c1(OC)c(C(=O)NC2CC(CNC(=O)C(C)(C)c3cccnc3)C2)csc1Cl c1(C(c2occ(C(=O)NCCCN(C(C)=O)CC)n2)NC)ccn2ncnc2c1 C(=O)(C(C(C)(C)O)NC(=O)CCC1CC(OC)C1)NC(C(CC)CC)C C1(C(N(CCCN(C)C(C2(c3cccs3)CC2C)=O)C)=O)CSCN1C C1(NC(CCNS(C)(=O)=O)=O)CN(C(C2(C)COC(=O)OC2)=O)CC1(C)C N1(C(=O)NCC(C)(C2CC2)OC)CC(C)(C(=O)OC)C(F)(F)C1 c1(C(=O)NC2CCC2NC(C2C3CCC2CC3)=O)scc2c1CCCC2 c1(OC)cc(C(=O)NC2CC(NC(C3CCC(C)(C)C3)=O)C2)cc([N+](=O)[O-])c1O C1(O)(C(=O)NCC2(O)CC(C(=O)NCC(=O)OCC#C)C2)CCSCC1 S(=O)(=O)(c1cccc(Cl)c1)NC1C(C)CN(C(=O)Cc2cccnc2)C1 c1(C(N2CCC(C(=O)NC34CCC(CC3F)C4)C2)=O)ccc2nccn2c1 C(CCC(C(=O)NC(C)CNc1cc(Cl)ncn1)NC(C)=O)OC n1(CC)c(C)cc(C(=O)NCC(O)Cc2cccc(F)c2)c1C CCC(CC)(CO)C(=O)N1CCN(C(=O)CCSCC(C)C)C(CF)C1 c1(C(=O)OC)ccc2c(c1)CCCCC2NC(=O)NC1CCC(=O)N(C)C1 CC1C(NC(C2CCC3(CC3)C2)=O)CCCN1C(c1nc(C2CC2)ncc1Cl)=O C12(C(N3CCN(C(CS(CC)=O)=O)CC3C)=O)CC(C)(C1)OC21COC1 Cc1ccc(C(=O)NC2CN(C(c3cnn(C)c3)=O)CC2C)nn1 Cc1cc(C(=O)NC2CC(C)N(C(=O)Cn3cc(C#N)cn3)C2)cnc1C c1(CC(N2CC(O)(C(CNC(C(Br)=C(C)C)=O)(C)C)C2)=O)cccnc1C C1(CNC(C2C(C)C2C)=O)CC(F)(F)CN1C(=O)C(O)Cc1ccc(F)cc1 c1(C(=O)NCCCc2nnc(C)n2C)cc(I)ccc1Br N(C(=NCC(C)C)NCc1ccoc1)CC1CCN(CC)C1 C1(CN(C(C2(CNC(C(C)OCOC)=O)CC2)=O)C)CCc2nccn2C1 CC1CCN(C(c2ccc(F)cn2)=O)C1C(N1CC(N2CCCC2=O)C1)=O c1(C(N2CCCC(NC(CCNC(COC)=O)=O)C2)=O)cc2n(c1)CCOC2 N1(C(C2(C(F)(F)F)CC(C)(C)C2)=O)CC2CN(C(=O)C(C)(C)F)CC2(C)C1 N1(C(C2CCC(=O)OCC2)=O)CCN(C(c2cnc(C(F)(F)F)o2)=O)CC(O)C1 C1(C)(C(=O)NCC(C)CC2CCCCC2)CC(O)CN1C(c1csnn1)=O Cn1cc([N+](=O)[O-])cc1C(=O)NC1CCOC(CNC(=O)C2CC2)C1 c1(OC)ccc(OCC2CC2)cc1.C(C)(C)(CC(=O)C1CCCC1)NCC1CC1 C1(Cn2cc(C3(F)CN(C(c4ccc(C(=O)NC)s4)=O)C3)nn2)CCC(OC)CC1 C1(C(=O)NCC(C)C)CCC2(CC2)N1C(=O)CC(C)(C)C1CCCO1 CCC(C(=O)NCC1CCC(NC(=O)CCC2CC(C)(C)CO2)C1)C(C)C O=C(C1CCc2nccn21)NC1C=CCN(C(=O)C=CCN2CCOCC2)C1 O=C(N=c1cc(Cl)[nH][nH]1)NNC(=O)c1cc(F)cc(F)c1 C1(NC(=O)CSC(F)F)CN(C(c2ccn(C3CC3(F)F)n2)=O)CC2(CCC2)C1 CCCCC(O)C(C)C(=O)N1CCC(CCC(N2CC3OC(=O)N(C)C3C2)=O)C1 C12(CNC(C3CCCC4CC34)=O)CC(CO)(CN1C(=O)C(O)c1ccsc1)C2 CC1CC(N2CCCC2)CN1C(C1CNC(=O)O1)=O N1(C(C(CC#C)O)=O)CC(C(=O)N(C)CCc2cnc[nH]2)CC12CCC2 N1(C(C)=O)CC2(NC(=O)C3=CCCCO3)CCC1C2 c1(C(N2CCC3(NC(c4cc(OC)ncc4)=O)C(C2)C3)=O)ccc(Cl)c(Cl)c1O C1(C(C)NC(c2cncc(C(F)F)c2)=O)CCN(C(=O)CCC2CCCO2)CC1 C1(Nc2c(C)c(N3CCCC3)ncn2)C2CC3CN(C(=O)N(C)C)C1C3C2 c1(C(=O)NCC(C)(C)NC(C2C3(CC3)C23CC3)=O)cc(N)c(F)c(F)c1Cl N1(C(CCCC(=C)C)=O)CCC(C)(C)CC1C(=O)NCc1ccc(F)nc1C C=CCCCCC(=O)NC1CCCCC1CNC(c1ccc(F)s1)=O CCCCC(CC)CC(=O)NC1C2CC1N(C(c1sc(C)nc1C)=O)C2C S(=O)(=O)(c1ccc(=NCC2OCCc3sccc32)[nH]c1)N1C(C)CS(=O)CC1 Cn1nccc1C(=O)NC1CN(C(c2nscc2I)=O)C1 c1(C(=O)NCC(C2CC2)NC(c2cc(C3CC3)ns2)=O)cc2c(nn1)OCCS2 C(N=c1nc(N2CCCC(CN(C)C)C2)c2c([nH]1)CCS2)c1ncc(C)s1 CC1CN(C(C(=O)NCCCF)C2CC2c2ccco2)c2cc(Cl)ccc2O1 c1(CC)ccoc1C(=O)NC1(CF)CN(C(=O)Cc2cnn(C(F)F)c2)C1 c1(CC(C)C)c[nH]c(C(=O)NCC2(O)CC(CNC(C3(O)COC3)=O)C2)c1 CC1CCC(Cl)=C(C(=O)NC(C2CCN(C(C3CC(C#N)C3)=O)CC2)(C)C)C1 C1(CN(CC(C)(C)OCC(=O)OC)C(C2COCC2CN)=O)CCC(F)(F)CC1 C(N=c1ccc2nnnn2[nH]1)C1C(NC(c2cnc(C)s2)=O)CCCC1 CC1CC(NC(c2ccc(O)nc2)=O)CN(Cc2ccc(Br)nc2)C1 N1(C(C2C(CC)CCC2)=O)CCN(CC)CC(C)C1.C12CCCC(C1)CC(=O)N2 C(CCC(=O)NC(C(=O)NCCc1cncs1)C1(O)CCC1)OCCOC C(C1CCOc2ccccc21)NC(=O)Nc1ncc(C)nc1 C1(C(N2CC(F)CC2CNC(C2(CC3CC3)CCCO2)=O)=O)CCS(=O)(=O)C1 N#Cc1c[nH]c2ccc(-c3nc(Cc4ccc(OC(F)(F)F)cc4)no3)cc12 N1(C(CC2CCC(=O)N2)=O)CC2(CCNC(C3CCCSC3)=O)CCC1CC2 C(CC(N=c1[nH]c(Cl)ncc1Cl)C(C)C)NC(C(C)SC)=O C(=O)(CCCCCNC(c1cc(C#N)cs1)=O)N1CC(CC(C)C)OCC1 C(CCCCN(C)C(C1(C#N)CC1C(F)(F)F)=O)NC(C(C)SC(C)C)=O C1(NC(COC(CC)C)=O)CC2CC(C1)N(C(c1nnn(C)c1C)=O)C2 N1(C(CC(=O)OCC)=O)CCC(C(F)(F)F)C(NC(C2(CF)CC2)=O)C1 N1(C(c2c(OC)csc2)=O)CC(N(C(=O)C(C)C(F)(F)F)C)C2(CC2)C1 C12(CNC(CC=CC(C)(C)C)=O)CC(CCO1)N(C(=O)C(C1(O)CCCC1)F)C2 c1(OCCC)ccc(Cl)cc1C(=O)NC1CCN(C(=O)C2=COCC2)C1C C(CCN=c1[nH]c(-c2ccc(C)nc2)cs1)c1ccc(OC)cc1 c1(CN2CCN(c3cccc(NC(CC=C)=O)c3)CC2)c(Cl)cccc1Br c1(CN(C)C(C2C(CNc3cnc(C(F)(F)F)cn3)CCC2)=O)cccc(N)c1F N1(C(C2(C)CC2(F)F)=O)C(CNC(C2CNC(=O)C2)=O)Cc2ccccc2C1 c1(CCNC(=O)CCNC(C2COCCOC2)=O)nccc(O)n1 C1(C2CN(C(=O)CC3CC4CCC3CC4)C2)(NC(Cc2ccc(C)cc2)=O)CC1 CN1CCCCC1CCC(=O)NC1CCC(NC(=O)CC2CC2C(F)(F)F)CC1 N1(C(CC=CCC)=O)CC2CC1CN2C(c1cccc(I)c1O)=O C(=O)(C(CC(C)C)N(C)C)N(CCNC(CCCC)=O)CC1CC1 C(=O)(CCCCCCNC(=O)Cc1ccc(F)nc1)N(CC(N1CCCC1)C)C N1(C(CCCN(C)C)=O)CCC2CC1CN(C(=O)CS(=O)(=O)N(C)C)C2 N1(C(C2NC(=O)OC2)=O)CCC(CO)(CNC(C2CCC(F)(F)C2)=O)CC1 C(C(=O)NC1CCN(C(=O)CCCc2cccs2)CC1)(C(C)C)NC(C)=O C1(NC(CNC(COC(CC)C)=O)=O)COc2ccc(OC(C)(C)C)cc2C1 c1(C(=O)NCC2CC(NC(CCC(=O)OCC)=O)C2)sc2nccc(C)c2c1C c1(OC)cscc1C(=O)NCCC1CCCN1C(=O)CC(=O)N(C)C C(=O)(C(C)CC(C)(F)F)N1CCN(C(CCC(=O)N(C(C)C)C)=O)CC1 c1(CC)nn(C)cc1CNC(=O)Nc1nccc(-n2nc(C)cc2C)n1 N1(C(C2CC(SC)C2)=O)CCOCC(NC(c2cccnc2C)=O)C1 N1(C(C(CC)C#N)=O)CC2(CCCN(C(=O)CCCC3CCCO3)C2)C1 O=S(=O)(c1ccc(NC2CCOCC2OC(F)F)nc1)NCc1ccnnc1 CC1(C)OC(=O)CC1CNC(=O)C(=O)NCc1csc([N+](=O)[O-])c1 c1(C(N(C)CC2CCCN(C(=O)C(F)OC(F)(F)F)C2)=O)ccc(C#N)cn1 C12(C(N3CCC(OCC(=O)NCCC4CC(F)(F)C4)C3)=O)CCCN(CC1)C2 c1(C(N(C)CC2N(C(CCN(C(C)=O)C)=O)CCCC2)=O)cc(Cl)n[nH]c1=N c1(C(N2CCC(C(=O)NCc3ccc(O)nc3)C2)C)ccc(F)cc1 c1(C(=O)OC)c[nH]c2ccc(CN3CCCC(O)C3C)cc12 CC(C)CC(O)C(=O)NC1C2CCN(C(C3(C)CCC(=O)NC3)=O)CC12 C(=O)(C(C)C(=O)N(C(C)CNC(=O)Cc1cncc(C)c1)C1CC1)OC CC1CCN(C(c2ccc(Cl)c(Br)c2F)C(=O)NC2(C)CC2)CC(C)O1 C1(C(=O)NCC23C(CN(C(C4(C)CC=CC4)=O)C2)C3)CC2CCC(C1)C2 c1(-n2cc(CNC(C3(COC)CCOCC3)=O)nn2)ccc(Cl)cc1Cl CCCN=C(NCCOc1cccc(F)c1)NCC1(F)CCOC1 C(=O)(C(CNC(=O)C(F)CC1CCOC1)CC1CC1)NC1CCC(=O)C1 c1(-c2[nH]nc(C(=O)NCCOC)c2Br)ccc2c(c1)C(=O)NC2 N1(C(C(C)C)=O)CCN(C(C2CCCCC2O)=O)C(C)C1 CC(C)CCN=C(NCC(N1CCN(C)CC1)C(C)C)N1CCCC(C)(F)C1 CC(CCN(C)Cc1cn(CCOC2CC(Cc3ccncc3)C2)nn1)C(=O)O c1(C(=O)NC(CN(C(=O)C=Cc2ccsc2)CC)C)cnc2n1C(C)CCC2 N1(C(C(CC#C)C)=O)CC2CCC(NC(=O)Cc3cccc(F)c3OC)(C2)C1 C(=O)(C(CCNC(c1cnn(CC)c1)=O)OC)N(CC=C)CC=C CC1CC(C(=O)NC2CCCC2CC(=O)NC(c2nncn2C)CO)CC(=O)N1 C(c1ccc(F)c(F)c1)=CC(=O)NCC12CC1CN(C(C1CC1C(F)F)=O)C2 C=CC1CN(C(C(=O)NC2CCOC2)C(C)C2CCOC2)CCO1 N1(C(N2CCCC(C)C2)=O)CCOC2CN(C(=O)Cc3ccc(Cl)cc3)CC12 C(=O)(C(CNC(=O)CC1CC1(C)C)CC1CC1)NC(COC)(C)C c1(C(=O)NCC(CNC(c2c(C)cc(C)s2)=O)C)ccnc(O)c1Br C(=O)(C1=CCCCCC1)N1C(CC(=O)N(C)CC2(CO)CCC2)C2CCC1C2 S(=O)(=O)(c1cc(Cl)cc(Cl)c1)N1C(C(=O)NCc2ccc(Cl)s2)C=CC1 C1(=O)C(CC)(CC)CN1.C1(C(C#C)OC)CC(=O)OC1(C)C.C12(C#C)CN(C1)C2 CC1(CCC(=O)NCCCn2cnnc2)CN(C(c2csnc2Cl)=O)C1 C(C)(CO)(C(=O)NCC(C)CN(C(=O)CCCc1csc(C)n1)C)OC C1(OCCNC(C=CC(C)(C)C)=O)CCN(C(c2csc(S)n2)=O)C1 C1(CCC(=O)NC2CCC(NC(c3nnn(C(C)(C)C)n3)=O)C2)C(=O)NN=C1C c1(CN(CCCC(OCC)OCC)C(C2CCCCO2)=O)cc([N+](=O)[O-])n[nH]1 S(=O)(=O)(c1cc(C)oc1C)NC1CCN(c2ccc(OC)cc2)C1 C(N(C)N1CC(O)(c2cccc(F)c2)C1)C1(CSC)CC1 N1(C(CC(C)(C)C(F)F)=O)CCc2ccccc2C(NC(C2CCC3CC23)=O)C1 O=S(=O)(c1ccc(NC2COc3ccc(F)cc32)c(F)c1)NCCCCC=CBr N1(C(COCC(=O)NC)=O)CCC2CCCC12CNC(c1coc(SC)c1)=O C1(Cc2cc(C(=O)NC(CN(CCCC)C)C)[nH]c2)CCC(n2ccnn2)C1 C=CC(C)(C)CC(=O)NC1(CO)CCN(C(C2(C3CCCCO3)CC2)=O)C1 N1(C(c2cn(CC)nc2C)=O)CCC2CC(NC(c3ccsc3C)=O)CCC2C1 C1(CNC(c2cc(Cl)cs2)=O)CC(C(F)(F)F)CCN1C(C1CCCSC1)=O Cc1noc2nc(C(N3CC(NC(c4c[nH]nc4F)=O)C(O)C3)=O)ccc12 CC(CN(C(=O)CC1CN(C(C2CN3CCC2C3)=O)CCO1)C)C(F)(F)F CC(CC(F)F)C(=O)NC1CN(C(c2c[nH]nc2C(F)F)=O)CC1(C)C C(c1ccc(O)cc1)=C1CN(C(=O)NCc2csc(N3CCCCC3)n2)C1 c1(C(N2CC(CCO)(NC(C(COC)CC3CC3)=O)C2)=O)cnn(C)c1OC N1(C(c2n(C(C)C)ccc2)=O)CC(CNC(c2cnc(Cl)s2)=O)C(C)(C)C1 C1(CC)CCCC(NC(C2(CNC(=O)CCN3CCCC3)CC(C)(C)C2)=O)C1 c1(-c2onc(Cc3ccc(C)cc3Br)n2)ccc2cncnc2c1 N1(C(CC2CC(CC)C2)=O)CC2CC2C1C(=O)NC1CCC2(CC2)C1 c1(CC(N2CC(NC(c3n(CC=C)ccc3)=O)C2)=O)cn2c(C)csc2n1 N1(C(CCNC(=O)NC)=O)CCN(C(c2cccc(-c3ccncc3)c2)=O)C(C)C1 CC1CCN(C(=O)COC2(C)CCC2)CC1CC(=O)N(CC(F)F)CC1CCC1 C1(CNC(COC2(C)CCCC2)=O)CC2CCC(C1)N2C(C1(C)CCNC1=O)=O C1(C)(CNC(CNC(C)=O)=O)CN(c2nc(C(C)C)cc(C)n2)CCO1 C1(CC)CCC(F)(F)CN1CCC#N.C12(CCCN1C(=O)OC(C)(C)C)C(=O)O2 C(=O)(CCCCO)Nc1scc(CC(=O)OCC)n1.C1(=O)C(=O)NCCCN1C c1(CC)cccc(NC(=O)C#CCNC(C2CCCC(C)C2)=O)c1F CON(CC1CC1)C(=O)C(c1ccoc1)N(C)C(c1cnc(N)cn1)=O c1(C2C(OC(C3(COC)CCCO3)=O)C2)c(F)cc(Br)cc1F C1(NC(C(C)NC(C(CC=C)(C)O)=O)=O)CC12CCCCCC2 c1(CC(=O)NC2(CNC(CCc3scc(C)c3)=O)CCOC2)c(C)noc1C N1(C(Cc2nnc(C)o2)=O)CCC(C)N(C(C2CC(=O)N(C3CC3)C2)=O)CC1 C#CCCCCCCCC(=O)NC(CNC(C1C(Cl)(Cl)C12CC2)=O)C(C)(C)C C(=O)(C#CC1(C)CCCO1)N1CCC(NC(c2c(O)ccc(OC)c2)=O)C1C CCC(C)(C)C(O)C(=O)N(CCC(=O)NCCc1c[nH]nc1O)CCCO C1(CC(=O)NCC2CC(OCC)C2)CN(C(=O)CCC2(C)N=N2)CC1C n1(CC(COCCOC)C)c(-c2cn(C)nn2)csc1=Nc1ccc(F)c(F)c1 c1(N2CCN(C)C(CNC(=O)CSC3CC3)C2)ccc2c(n1)CC(C)(C)CC2=O N1(C(CC(C)P(C)(C)=O)=O)CCCC12CCN(C(=O)C(C)(F)F)C2 c1(C(=O)NCC2OCCC(NC(C(CC)(C)C)=O)C2)cc(C#N)oc1C c1(C(N(C(C)C)CCO)=O)cc(-c2ccc(F)nc2F)cn2ccnc12 N1(C(CCCC)=O)CCC2C(CCCN2C(C2CN(S(N)(=O)=O)C2)=O)C1 c1(C(c2n(CCCOC)nnn2)NCC(Cl)Cl)c(Cl)ncn1C C12(NC(c3cc(CC)nn3C)=O)CCC(C(=O)NCC3CCC(C)C3)(CC1)C2 CC1CN2CC1(C)SCC2=O.N1(CCNC(C2(C(N)=O)CC2)=O)CCS(=O)CC1 C1(C(=O)N(CCn2c(C)ncc2)CCO)CCCN(CCC2CC3CCC2C3)C1 N1(CCOCC)CCCC(NC(c2c[nH]nc2CC2CCC(OC)CC2)=O)C1C N1(C(=O)CCc2cccc(F)c2F)CCCN(C(=O)NC(C2CC2)C2CC2)CCC1 Cn1ccc(C=CC(N2CC(O)CC2CC(=O)NCCN(CC(C)(C)C)C)=O)c1 c1(C(N2CC3N(C(C(C)OCOC)=O)C(CC3)C2)=O)cc2ccccc2nn1 c1(C(N2CC3(CC(NC(C(c4n(C)ccc4)=O)=O)C3)C2)=O)cc2n(n1)CCCO2 C1(C(F)(F)F)CC2(CN1)CC2(F)F.CC1C2CC(C(=O)C(Cl)(Cl)Cl)(C2)N1C=O CC(C)C(C(=O)NC1CC(C)(NC(c2ccc(CO)nc2)=O)C1)c1cnn(C)c1 C1(OCCOC)CCC(c2nc(Cc3cccs3)nn2CC(C)(C)O)CC1 C1(N(C(=O)CCc2cnc[nH]2)CC)CC2CC(C1)N(Cc1cnn(C)c1)C2 C1(C(=O)NCC(C(=O)N(C(C)CC2CC2)C)OC)CCOCC1(C)C c1(C(=O)NC2C(NC(CC(n3ccc(C)n3)C)=O)CCC2)ccc2scnc2c1 c1(C(=O)NC(CN(C(=O)CC2(c3ccon3)CC2)CC)C)nc[nH]c2ncnc1-2 N1(C(=O)NCC2(C(=O)NCC(O)CCOC)CC(=C)C2)CCOCC1=O c1(C(=O)O)ccc(F)c(CN(C=O)C(C2(c3cc(Cl)cc(Cl)c3)CC2)=O)c1 CC(C)C(C)C(C)CC(=O)N1CCOC(CNC(=O)C=Cc2cncs2)C1 N1(C(C2CC(NC(C(C)CC3CCC3)=O)C23CCC3)=O)CC2COCC2(C)C1 C=C1CCC(C(=O)NC2C=CC(CC(=O)NC3(C)CC(F)(F)C3)C2)CC1 C1(NC(C=CC=CC)=O)CC2CN(C(c3cc4cnccc4[nH]3)=O)CC2C1 c1(C(=O)OC)ncccc1NCC(C(=O)CC1CC1)NC(=O)OC(C)(C)C C1(CC#C)(C(=O)N(CCCNC(=O)CC2CCC23CCC3)C)CCCOC1 N1(C(=O)NC(c2cnn(C(C)C)c2)CSC)CC(O)C(O)C12CCCC2 C(=O)(CCC(C)(C)C)NCCN(C(=O)CC1C(=O)ON=C1C)CCOC N1(C(C(COC)Cl)=O)CC(NC(c2ccc(Br)cc2Br)=O)C2(CC2)C1 C1(C(=O)NCC2(F)CN(C3(CC)CC3)C2)(COCC)CCCCC1.C12(CC1)C(=O)N2 N1(C(C(C)CO)=O)CC2(CCN(C(=O)Cc3c(Cl)cnn3C)CC2)CC1C C=C1CCN(C(c2cc(C(N)=O)co2)=O)C(C(=O)NCC2CCCCO2)C1 c1(CCN2CCC(n3cc(C(N)=O)nn3)CC2)cc(F)cc(Cl)c1 c1(OC)ccc(C(N2CCCC(NC(c3ncnn3C)=O)C2C)=O)cc1Cl C(CCC(F)(F)F)(C(=O)OCc1ccc(-c2ccccc2)cc1F)OC C1(NC(c2n(CCC)ccc2)=O)CN(C(=O)C(C)Oc2ccccn2)CCC1C c1(OC)cc(OC)nc(N2CC(CNC(=O)CC(C)(O)C3CC3)CC2C)n1 C=CCC(C)(C)C(=O)N1CCC(C)(CNC(=O)C(c2ccc(F)cc2)C2CC2)C1 c1(C(=O)NC(C2CCN(C(CNC(C)=O)=O)C2)C)cnc2ncnn2c1C(C)C C(=O)(CCC(CC)NC(=O)CC1CCC(=O)C1)N1CCC(C(C)(C)C)CC1 C(=O)(C1=C(Cl)CCC1)N(CCOC1CCN(C(C2C(CCC)CCC2)=O)C1)CC C(O)(C(F)(F)F)C1(C(=O)NC(C(C)NC(=O)CN(C)C)C)CCC1 CN1CCOC(C(=O)NCC2(O)CCN(C(=O)C=C(C3CC3)C3CC3)C2)C1=O Cc1c(N(C(c2ccnc(Cl)c2)C(=O)NCC(C)C)C)cccc1Cl CC(O)CCN=c1ccnc(N2CCc3ncncc3C2)[nH]1 N1(C(c2cc(C(C)=O)oc2)=O)CC2(CCN(C(C3CCC(C)O3)=O)C2)C1 C1(Nc2ncc(C)cn2)CC12CCN(C(c1cc(C3CCOCC3)on1)=O)CC2 C1(C(=O)OC)CN(S(C)(=O)=NC(=O)C(C)C2(O)CCN(C3CC3C)CC2)CCO1 C1(CNC(c2cn(CCOC)nc2)=O)CC2(CCC2)CN1C(=O)CCC(F)F C1(CNC(c2nnc(C)s2)=O)CC2(CCN(C(c3ccc(=N)[nH]c3)=O)C2)CO1 n1(CCOC)ccc(C(=O)NCC2CC2NC(=O)C(C)N(CC(F)(F)F)C)n1 Nc1cc(F)c(O)cc1C(=O)NCC1CCCCN1C(=O)CSCC1CCCO1 c1(C(=O)NC(CNC(CC(CCC)O)=O)C)ccc2nc(O)[nH]c2c1F c1(C(=O)NC2C(CNC(C(C)OC)=O)C2)cnc(C)nc1C1CC1 Cn1cc(-c2csc(C3CC3C(N3CC(=O)NC(C)(C)C3)=O)n2)c2ccccc12 c1(NCC(C)O)ccc(S(=O)(=O)N2CCCCC2C2CCOCC2)c(Br)c1 n1(CC)cc2ccc(C(=O)NC3CCC(NC(C4(OC)CCOC4)=O)C3)cc2n1 C1(C(N(C(C)CN(C)C(c2c[nH]nc2C(F)F)=O)C)=O)CCC(C)(C)CO1 CC1(C)CC(C(N2CC(C)(NC(=O)CC3CCOCC3)C2)=O)CC(C)(C)O1 c1(C(=O)NCC2CC2NC(C2CS(=O)C2)=O)cc2cccn2cn1 Cc1ccc(C(=O)NCCCC(O)C(=O)NCCC2CCC2)cc1C C(=O)(C(C(C)(C)C)NC(=O)CC1CC(C)(C)CO1)NCC1(C)N=C(C)SC1 c1(C(=O)NC2CC(NC(c3ccc(C#C)o3)=O)C2)cnc(C)c(C#N)c1 Cc1cc2c[nH]nc2cc1-c1nc(C2(C)CC3(CC3)C2)no1 C1(CNC(C2N(CC)CCCC2)=O)CC2(CO1)CN(C(=O)C(CC)(CC)CO)C2 C1(NC(=O)CCOC2CCCCC2)CCCC12CN(C(c1cn[nH]c1)=O)C2 c1(SCC(CNC(=O)CSC(F)F)OC)nc(-c2ccccc2)no1 C(C(C)(Cn1cccn1)NC(c1n[nH]cc1Cl)=O)NC(CC1CC(C)C1)=O Cc1[nH]nc2ncnc(N3CC(C(C)NC(=O)CSC4CCCCO4)C3)c12 c1(C(=O)NC(C)C(CO)NC(c2nccnc2N)=O)ccc2nonc2c1 C1(C(CC)C)CCN(C(=O)C(C)NC(=O)C(C2CCCCC2)F)C1 N1(C(c2c(C)ncs2)=O)CCC(C(F)CNC(=O)CN2CCCC2CO)CC1 C1(CC(=O)NC(C(C)O)C(=O)OC(C)(C)C)(C(F)(F)F)CC(=O)N(O)C1 C1(C(=O)NC(C)CNC(=O)CC=CCN2CCCCC2)COC(=O)N1C C1(C(=O)NC2(C)CCCN(C(C3N(CC)CCC3)=O)C2)Cc2ccccc2CO1 C(C)(N=c1[nH]ncs1)C1OCCN(C(C)C(C(=O)CCCCN(C)C)=O)C1 CCC(CN(C)C)CC(=O)NCC1CC(NC(=O)C(C(C)C)NC(C)=O)CCO1 C1(C(N(C2CC=CC2)CC)=O)CCOCCN1C(=O)CC1CC=CC1 N1(OC(C2C(C)C2)=O)CCCC(CO)CC1.N12CCCC1(C)CC=CC2=O N1(C(=O)C(F)=CCCF)CCC2(CC1)CN(C(c1cc3c(nn1)CCC3)=O)C2 CN1CCN(c2cc(C(=O)N(C3CC3)Cc3nn(C)cc3I)on2)CC1 C(=O)(C#CC1CCC1)N(C1CCN(C(=O)COc2ccc(C#N)cc2)C1)C c1(OCC)ccc(CCC(=O)NCC(C2CC2)NC(C2CC23CC3)=O)cc1 CCC(C)(CNC(c1conc1C(C)C)=O)C(=O)NOCC(F)F C1(C(=O)NC2(CC=C)CCOC2)CC(C)(C)CCN1C(=O)Cc1nc(C)c(C)[nH]1 O=C(CCC(CF)CF)NC1CC2CC(NC(C3CN(CC(F)(F)F)C3)=O)CC21 c1(NC(C2(NC(C3CC4(CC4)CO3)=O)CC(F)(F)C2)=O)ccc(O)c(F)c1 N1(C(COC(Cc2cn(CC)nn2)=O)=O)CCCCC1c1n[nH]cc1C(=O)NC CS(=O)(=O)C1(c2nnc(N3CCC(F)(F)CC3)n2CC2CCCO2)CCNC1 N1(C(c2oc(C(=O)OC)c(C)c2)=O)CC2CCC2(CCNC(C2(C)CC2)=O)C1 CCC(F)(C(=O)OC)C(=O)N1C2CCC1C(CNC(=O)COc1cccnc1)C2 CC1(CNC(c2ccc(-n3cnnn3)cc2)=O)CC(F)(F)CN1C(C1CCC1)=O C1(C(N(C(C)C)CCNC(C23CCCC2C3(F)F)=O)=O)CCCCN(C)C1=O C1(NC(Cc2c(C)non2)=O)CCCC(CNC(=O)CCCN(C)C)C1 C(=O)(CCCCCS(N)(=O)=O)NC(C)Sc1ccc(CO)cc1 N1(C(c2ccc3cccnn23)=O)CCC2(CCCN2C(C2CCCS2)=O)C1 C(=O)(CCCC1CC1)N1CC(C(C(=O)N(C(C)CO)CC2CCC2)O)C1 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)CO)CC1C C1(C(=O)NC2C(CNC(Cc3c(C)scc3)=O)COC2)Cc2ccccc2S1 Cc1cc(C(=O)NCCC(C)N(C)C(c2cc(CO)n(C)n2)=O)cnc1O c1(N2CCC(C)(NC(C(C3CCCOC3)OC)=O)C2)ccncc1C#N CCC(CC)CC(=O)N1CCN(C(c2cncnc2)=O)C(C(C)(C)C)C1 c1(C(N2C(C)CC(NC(=O)CC3(O)CCOCC3)CC2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(OC)cc(C(N2CCC(NC(=O)CCn3cc(C)cn3)C(F)C2)=O)c(F)cn1 N1(CC(=O)NCCn2cc(Cc3cocn3)nn2)CCCCC1=O C1(NC(c2ccns2)=O)CC(C)C12CCC2.C1(CC(=O)NCCOC)(COC)CC1 N1(C(CCNC(=O)NCC)=O)CC=C(C(=O)NC2(CC3CC3)CCC2)C1 c1(OC)cc(C(=O)NC2CN(C(c3cnc(C)[nH]3)=O)CC2C)cc(C2CC2)c1 Cn1cc(C(=O)NCCC2CN(C(c3ccnc(C4CC4)n3)=O)C2)cc1Br Cc1cc(C(=O)NCC(O)CN2CCCC(C(N)=O)C2)nn1C(C)C C1(C(N2CC(C(C)NC(C(c3ccccc3Cl)C)=O)C2)=O)CCCC(C#N)C1 c1(C(=O)NCC2(F)CN(C(C3C(C=C)C3)=O)C2)ccc(C)c(Br)c1 c1(OCCN(C)CC)ccccc1-c1cn(CCC2C=CCCC2)nn1 C12(C(=O)OC(C)(C)C)C(NC(c3ccn4ccsc34)=O)C3CC1C2C3 n1(CC(=O)NC(CC=C)CNC(C2CC(=O)NC2(C)C)=O)c([N+](=O)[O-])cnc1C C1(CCOC)(NC(c2cnccc2C)=O)CCN(C(c2nocc2Cl)=O)C1 Cc1cc(C)c2c(Cl)c(NCC(=O)OC(C)(C)C)sc2c1 N1(C(C(=O)NCC(F)F)=O)CCC2(CC1)CC2C(=O)NC1CCCC1C1CC1 c1(NC(N(c2cn(C)nc2)CC2CC2)=O)cc(C(F)(F)F)ccc1O c1(C(=O)NC(C(=O)N(CCCCC=C)C)C)ccc2c(c1)CCC2 C1(CCNC(=O)CCCF)CN(C(=O)COCc2cccc(Cl)c2)CCO1 c1(CN(C(=O)Cn2ccccc2=O)CCCNC(COC)=O)ccc(C)cc1Br N1(C(c2c(Br)ccc(C)n2)=O)CC2CCC1CN2C(=O)CC(O)C(C)C C1(NC(C(C)N(C)C)=O)CCC2(CC1)CN(C(c1n[nH]c3c1COCC3)=O)C2 C1(NC(C2CC(=C)C2)=O)CN(C(c2c(N)cccc2Cl)=O)CCC12CCOCC2 N1(C(C(CCCC)C)=O)CCCC2CN(C(c3ccc(=O)n(C)c3)=O)CCC12 c1(C(=O)OC)nc(N2CC3CC3C2)c2c(n1)CCC(Nc1ccccc1)C2 Cc1nc(Cl)ccc1CC(=O)NC(C)CNC(=O)CCCNC(C1CCCC1)=O N1(C(CCCNC(=O)OC)=O)CCCC(F)(C(=O)NC2COCCC2O)C1 c1(CC(=O)NC(CC=C)CN(C(=O)CCC(=C)C)CC)coc2cc(O)ccc12 C1(C)(C(=O)NC)CCCN1C(=O)CC1CCN(C(c2cn[nH]c2)=O)C1 CC(CN=c1[nH]c2c(c(=NCC3CN(C)CCN3C)[nH]1)COCC2)c1ccncc1 N1(CCNC(=O)C=CCC2CCCO2)CCN(C(C2CCNC(=O)C2)=O)CC1 O=C1CS(=O)(=O)CC(C(=O)NC2CC(NC(c3c[nH]cc3Br)=O)C2)N1 C=CC1COCCN1C(=O)CCOC1CCCC(O)C1.C12CN(C1)C2=O c1(C(=O)NC2(CCCC)CC2)cc(CNC(=O)C=CCN2CC2C)nn1C c1(OC)ncccc1C(N1CC(C)C(C)(CNC(=O)CC2CNC(=O)C2)C1)=O C(C(O)CCCC)NC(C(C1(O)CN(C(CCOCC#C)=O)C1)F)=O C1(OC)CCC(c2cn(CCCCNC(=O)CCCC3CC3C)nn2)CC1 c1(OCC(=O)NC2C(NC(c3cncc(CC)n3)=O)CC2)ccc(Cl)cc1C CC(C)(CCNC(=O)CC1CCC(O)C1)NC(C1CC(N(C)C)C1)=O C1(C)(CC)CCCN(C(C23CC(CN2C(c2ccc(C)cc2OC)=O)C3)=O)CC1 C1(C)(NC(c2c(OC)cccc2)=O)CC(O)CN1C(=O)C1=C(Cl)CCC1 N1(C(F)(F)F)CC(N=c2ccnc(N3CCCCC3)[nH]2)C1.c12ccccc1S2 CC1CCC(C(=O)N(CC(C)CNC(c2nn(C)cc2Cl)=O)C)CC1 C12(NC(c3ncccc3Cl)=O)CCN(C(c3cncc(C(F)F)c3)=O)CCC1C2 C(=O)(C#CC1CCC1)N1C(CNC(C2C(C)(C)CCO2)=O)CCCC1 c1(C(=O)NCC2CN(C(c3ccc(C)s3)=O)C3C2C3)cccc2nn[nH]c12 C1(C(=O)NCCn2cnnc2)(CC)CN(C(=O)C(N)=O)C1 C(CN=c1ccc(Br)c(OC(F)F)[nH]1)=CCC CC1C(N2CCCCC2)CCN1C(=O)Cn1ncccc1=O C1(C(C(=O)NCc2ccc(CC)s2)(C)C)CCCN(C(=O)C=CCO)C1 C(=O)(C1=CCCC1(C)C)NCCC1CCN(C(C2C(C(=O)OCC)CCO2)=O)C1 C1(C(=O)NCC=CCNC(c2c(CO)cn(C)n2)=O)CC(=O)NC(=O)C1 c1(C(=O)NC2CC(CNC(Cn3c(C)nnn3)=O)C2)cn(C(C)C)nc1C c1(CC(=O)NC2(CC)CN(C(COCCC#C)=O)C2)ccc(C)c(F)c1F Cc1onc(Cl)c1C(=O)NC(C)CNC(c1nccn1C(C)C)=O N1(C(CCSCCCC)=O)CCC(C)(NC(C2CCCC2(C)C)=O)C1 C(=O)(C(CCF)NC(c1cc(OC)n[nH]1)=O)NC(C#C)CC c1(C(C(=O)NC(CC)CNC(c2cn(C)nc2Cl)=O)(C)C)cccc(Cl)c1F N1(C(Cc2nnc(C)s2)=O)CCCOC(CNC(c2ccnc(C(C)C)n2)=O)C1 Cn1nc(C(=O)NC2COCC2NC(C2CC23CCC3)=O)c(C(F)(F)F)n1 C1(O)(COC)CCCN(C(c2cnn3ccn(C)c23)=O)CC1 N1(C(c2nccc(OC)c2)=O)CCC(NC(C2CCCC2(C)C)=O)CC(O)C1 C(=O)(CC1OCc2ncccc21)N1CCC(CNC(C(C)C2CCCC2)=O)CC1 CCC(F)(F)C(C)(C)NC(C1(NC(=O)Cn2cnc(=N)[nH]2)CSC1)=O Cn1nc(-c2cncc(Br)c2)c2c1CCN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 N1(C(C=C(CCC)C)=O)CCC(C)C(CC(=O)Nc2cnccc2C2CC2)C1 N1(C(C(=C(C)C2CC2)F)=O)CC(OC)CC(NC(c2ncoc2C(F)(F)F)=O)C1 N1(C(C(C(C)C)CN(C)C)=O)CC(C(=O)NC(C)(C)CF)C2(CCC2)C1 C=C(C)c1cn(CCC(=O)N(CC)Cc2coc(-c3ccc(Cl)cc3)n2)nn1 c1(C(=O)NC2CN(C(c3cc(C)nc(C)c3)=O)CC2C)cccn2ccnc12 c1(C(=O)NC2CCN(C(=O)CC3(O)CCCC3)CC2)cnc2[nH]c(O)nc2c1 CC1(NC(c2cn(C3CC3)nn2)=O)CCCCC1C(=O)NCCCC1CC1 C(C)(CNC(=O)C(=O)NC(C)C)(C(C)C)NC(C(c1ccc(OC)cc1)CC)=O c1(OCC)cc(C(=O)N(CC(C)CNC(C23CC(C)C2C3)=O)C)ccc1C N1(C(c2c(CC)cco2)=O)CC(F)(F)CC1CNC(=O)CCc1nc(C)c(C)[nH]1 c1(NC(c2c(-c3cc(C)ncc3)c[nH]n2)=O)cc([N+](=O)[O-])c(F)cc1Cl C(=O)(C(O)C1=CCCCC1)N1CC(OCCC(=O)NC2CC(=O)N(O)C2)C1 O(NC(=O)C(Cc1cc[nH]n1)NC(c1ccn(C2CC2)n1)=O)CC(CC)C C(=O)(C(O)CC(F)(F)F)N1CC(N(C(=O)C=CC2(C)COC2)C)C(O)CC1 C1(NC(C(c2cccs2)NC(c2cc(CC)on2)=O)=O)CN(C)NC1=O c1(C(N(C)CC2OCCN(C(C3(C=C)CC3)=O)C2)=O)cc2ccccc2cn1 C(=O)(CCCCCF)C(=O)OC.c1(C(N(CC#C)CC)=O)cc(CCN)on1 c1(OCC)cccc(C(=O)NCC23CCC(C2)N(C(c2cscn2)=O)C3)c1N C(=O)(C(F)(CNC(=O)C(C)C(F)(F)F)C(C)C)NCc1ncc(CC)s1 CCC(CC(=O)N(CCCNC(c1cnc(C(N)=O)cn1)=O)C)C(C)(C)C S(=O)(=O)(c1cc(C2C(CNC(c3cc(C)[nH]n3)=O)CC2)c(C)o1)N(CC)CC N1(C(C2C(C)C2)=O)CCOC(CCCNC(c2ccnn2C2CCOCC2)=O)C1 C1(NC(c2sc(C)c(O)n2)=O)CN(C(=O)CCc2nc(O)n[nH]2)CC12CCC2 Cc1[nH]nc2ncc(C(N3CCCCC3CNC(C3(C)CCCCC3)=O)=O)cc12 c1(C(=O)NCC(CC)NC(=O)CCC2CCCC2)cc(F)c(F)cc1Br c1(C(N(CC(CNC(C2(CC)CC2(F)F)=O)(C)C)C)=O)cccc(C(C)(F)F)c1 c1(OC)nc(C)ccc1C(=O)NCC1CC(C)N(C(c2c[nH]nc2C2CC2)=O)C1 c1(C(=O)NCC2(CO)CC2C(F)(F)F)nc(Br)n2c1CCCCC2 C1(CNC(c2cnc(O)s2)=O)CC12CCN(C(=O)COc1ccon1)CC2 C1(COC)(CNC(c2cc(OC)ns2)=O)CCCN1C(C12COC(C1)C2)=O N1(C(CNC(CCC)=O)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC2C1 C(=O)(C(C)(CC)C(=O)NC1CC(CNC(=O)Cc2cc(F)cc(Cl)c2)C1)OCC C(=O)(CCCN=[N+]=[N-])N1C(CC=C)(C(=O)NC(CN(C)C)C(C)C)CCC1 C12(C(=O)NC(C3CCN(C(=O)CCC(N)=O)C3)(C)C)CCC(C)(C1)OC2 C1(NC(=O)C(O)Cc2cnc[nH]2)CCOC12CCN(C(=O)C(F)F)CC2 c1(CCC(=O)N(CC(C)CSc2nccn2C)C)ccc(O)cc1 C=CCCCNC(C1C(C(=O)N)C1)=O.C(C(C)(C)C)OC(N)=O.C12(CC1)C(=O)N2 C1(CNC(CCn2c(C)csc2=O)=O)CN(C(c2cn(C)cn2)=O)CC12CC2 CCCCC(O)C(=O)N(C)CCNC(C1(F)CC1(F)F)=O CCC(C)C(O)CC(=O)N(CCCCCC(=O)N(C1CC2(CCC2)C1)C)C Cc1oc(C#N)cc1C(=O)NC(Cc1cnc[nH]1)C(=O)N(C(C)C(=O)OC)C c1(C(=O)NCC2CC2CNC(C2COCCO2)=O)ccc(Cl)cc1C(F)F c1(C(=O)NC(C)CN(C(=O)CSc2ccccc2)C)ccc2c(c1)CCN2 CCCC(C)CCCC(=O)N1CC(NC(c2ccnc3c2CCC3)=O)C(C)(C)C1 Cc1nnc2n1CCN(C(C1CSCCN1Cc1ccc(O)c(O)c1O)=O)C2 c1(C(N2CC(CNC(CCCCCC)=O)OCC2)=O)cc2n(n1)CCOC2 Cc1c(Br)cc(C(N2C3CCC(C3)C2C(=O)NC2CC(F)(F)C2)=O)cc1[N+](=O)[O-] C1(NC(C(C(CC)C)O)=O)CC2(CCN(C(c3ccn(CC(F)F)n3)=O)CC2)C1 Cc1nn(C)c(C)c1CC(=O)NC1CC(N(C)C(C2C=CCCC2)=O)C1 C(=O)(C1=NOC2COCC12)NCCC(CC)(C)NC(C1CON=C(C(F)F)O1)=O C1(NC(COC(C)C)=O)CC2CCCC(C1)N2C(c1c(Br)nnn1C)=O Cc1c(C(=O)NCCNC(=O)C(C)(C)N(S(C)(=O)=O)C)cccc1F N1(C(=O)OC(C)(C)C)CCC(CCN2CC3CC3(c3ccc(Br)cc3)C2)CC1 C(=O)(C(C)CC(F)(F)F)N1C2CN(C(c3c(-c4cc(C)no4)ocn3)=O)C(C2)C1 N1(C(CC(CC)C)=O)CCN(CC23CC(C(=O)OC)(C2)C3)CC1Cc1ccccc1 C1(C(=O)OC)C=CCCC1NC(C1(CO)CCOCC1)=O c1(C(N2C(C(=O)NC3CCCC(O)C3)CC(C)C2)=O)ccc2c(c1)CC2 C1(OC)CN(C(=O)CCOC)CC1CNC(C1(CCOC)CC1)=O.C1(C)CCC1 c1(C(N(CCCN(C(CC(COC)C)=O)C)C)=O)cnc(C2CCCC2)[nH]c1=N C1(NC(C2N(CC)CCC2)=O)CCN(C(c2ccccc2OC)=O)C(C2CC2)C1 CCCC(CC)CCC(=O)N1CCC(C2(C)CC2)C1.C1C(C)(C)CC(=O)N1 C(=O)(C(CCCOC)NC(c1[nH]nnc1C)=O)NC(c1nn[nH]n1)CC C(=O)(C1CCc2cccc(F)c21)N(CC1=NOC2CN(C(C3(C)CC3)=O)CC21)CC C(=O)(C1=NOC2COCC12)NCCCCCNC(=O)CSc1cn[nH]c1 c1(N(C)C)cc(F)ccc1C(=O)NCC1CCN1C(C1(C2CCCCO2)CC1)=O c1(CC)nccn1C(C)CC(=O)NCCCCN(C)C(C1(C)CCC1)=O c1(C(=O)NCC2N(Cc3nc(C)on3)CCC2)csc(C#N)c1 C1(NC(c2c(CC)ocn2)=O)C2CC3C(C2)C13C(=O)NC(C1CC=CCC1)CO C12(C(N3CCC(NC(CCC(CC)C)=O)(CC)CC3)=O)CC1Cc1c[nH]nc12 N1(C(=O)C(F)n2ccnc2)CC23CCCC2(C1)CN(C(C12CC1C2)=O)C3 CC1COC2(CCN(C(c3cncs3)C(=O)Nc3ccc(Cl)cc3F)CC2)O1 CC(C(=O)NCCC(C)(C)NC(=O)C(c1ccc(F)cc1)=O)C(F)F C(=O)(C(F)(F)C(F)(F)F)NC(C(C(C)C)C)CNC(C1CCCN1C(N)=O)=O c1(OCC=C)c(C(=O)NCC(C)(O)CNC(=O)C(C)SC(C)C)cccc1C c1(OCC(=O)NCCCCCNC(c2cnc(C)n2C)=O)cccc(F)c1F Cc1ccc2[nH]nc(C(=O)NC3CCN(C(=O)CC4CC=CC4)CC3CO)c2c1 n1(CC)ncnc1CNC(=O)C(C1(O)CCC1)NC(=O)CCCNC(N)=O C1(CN(C(c2cc(SC)oc2)=O)C)CCCN(C(=O)CC(O)CN(C)C)C1.C1CC1 C12(NC(CCCc3onc(C)n3)=O)CCC1CN(C(c1cccc(C)c1O)=O)C2 CC1CN(C(=O)CCc2ccc(CO)cc2)CCC1NC(C1C2CCC1CC2)=O C1(C(N2C(C(=O)NCCn3c(CC)nnc3)CCC2)=O)CC(C)CCO1 CC1(C)CC(O)(C(N2CC(CNC(c3ccc(C(F)F)cc3)=O)C2)=O)C1 Cc1nc(C(=O)N(C2CCCN(C(c3cccc(SC4CC4)c3)=O)C2)C)c(C)s1 N1(C(c2ccc(C)nn2)=O)C2CCC1C(NC(c1scnc1C(C)(C)C)=O)C2 N1(CC(=O)NC(c2ccccc2F)CNC(C2(C)CC2F)=O)CCS(=O)(=O)CC1 C=CCC(CC=C)C(=O)NCC(O)C(F)(F)F.C1C(=O)N1C CC1CC(NC(c2cc(O)n(C)n2)=O)CCN1Cc1ncc(Cl)n1C N1(C(CC=CC=C)=O)CC(C(N2CCC3CCCC23)=O)CC(C)(C)C1.CC C1(O)(CN(C(=O)Cc2cc(Cl)cs2)C)CCN(C(C2CCCCC2O)=O)CC1 C(=O)(C(O)C(C)NC(=O)Cn1ccc(C)c1)NC1(COC)CCC1 n1(C(C)C)cc(C(=O)N(C)CC2CN(C(=O)C(C)C3CC3)C2)cn1 C1(CNC(c2ccc3c(c2)CCCC3)C)CC2CCCCN2C1=O C(C(=O)N=c1ccn(C(C)(C)C)[nH]1)(C(C)(C)C)NC(c1c(C)ccs1)=O c1(C(C(=O)NC(CC)C)N(CC)Cc2cccc(F)c2C)cnc(OC)c(C)c1 C#CCCCC(C)C(=O)NCCC1CC(NC(=O)COCC2CCCOC2)C1 c1(C(C(N)=O)NC(C2CC2c2cn[nH]c2)=O)cccnc1 c1(C(=O)NCC(CO)NC(C(c2cccs2)SC)=O)cc(COC)cs1 C1(C(=O)OC)(OC)CC(O)C1.C12(CCOC1)C(=O)N2.C(=O)(C(C1CCC1)OC)NC C(C(C(=O)NCC1CC(NC(=O)CNC(=O)C(F)(F)F)C1)N(C)C)N(C)C C(=O)(CC(C)(C)C(F)(F)F)NCC1CC(CNC(CCC(=O)OCC)=O)OC1 N1(C(c2cccc(C)c2Cl)=O)CCC(C2CN(C(=O)C(F)C(C)C)C2)CC1 C1(C(N(C2CCCC2)Cc2ccccc2)=O)CCC(NCC(C)O)CC1 c1(OC)cnc(F)c(C(=O)NCCC2(O)CCCN(C(c3ccnnc3)=O)C2)c1 N1(C(C2N(C)C(=O)CC2)=O)CCC2(CC1)CC2(C)C(=O)NC(C1CCC1)C1CC1 c1(-c2n(-c3c(C)cc(F)cc3)nc(-c3ccoc3C)n2)ccc2ccccc2n1 C1(NC(C2(C)N(C(c3c(OC)ncc(Br)c3)=O)CC2)=O)CCC2(CC1)OCCO2 C1(C(N(C(C#C)C)CCCC)=O)CN(C(c2cc(F)ccc2C)=O)C(C)(C)C1 c1(C(N2CC3CN(Cc4cccc(I)c4)C3C2)=O)ccc(F)c2cccnc12 N1(C(C(=O)NCCOC)C2CC2C(=O)OC)c2ccc(Br)cc2CC1C c1(NC(c2ccc(F)cc2)CC)ncccc1S(=O)(=O)NC(C1CC1(C)C)CO C1(CC)CN(C(c2ncn(C)c2C)=O)CCC1NC(=O)CCc1cccn1C C(=O)(CCCCCF)N1CCC(CN(C(c2c(OCC)oc(C)n2)=O)C)C1 N1(C(C(C)O)=O)CC(NC(c2cnc(-c3ccccc3)o2)=O)CC2(CC2)C1 c1(C(=O)NCC(CC)Nc2ccnc(C(C)CC)n2)ccnc2ccnn12 C(=O)(C#Cc1ccccn1)Nc1ccc(SCC)cc1C c1(C(=O)NCC2C(NC(C(C(=C)C)(C)C)=O)CCC2)cncc2cnccc12 N1(C(c2cnn(C(F)F)c2)C(=O)NC2(C)CC2)CCc2c(Cl)cccc21 c1(C(=O)NCC2CN(C(C(Cc3cccc(OC)c3)=O)=O)C2)cccc(O)c1C c1(OCC(=O)NCCCN(C)Cc2c[nH]nc2C(C)(C)C)cccnc1 C#CC1(C(=O)NCCCC(CO)NC(=O)CC2CC(C)(C)CO2)CCCC1 C1(C(=O)NC2C=CCN(C(c3ccc(C#N)s3)=O)C2)CC12CCS(=O)(=O)CC2 CC(C)S(=O)(=O)c1ccc(C(N2CC(F)C(O)C2)=O)cc1 C(C)(c1ccccc1OCCSC)=CCN1CCN(C(C#C)CC2CCCO2)CC1 C1(NC(C2OCC(C)C2)=O)CCCCN(C(c2cnn(CCO)c2N)=O)C1 Cc1onc(C2CC2)c1C(N1CCCCC1CNC(c1ccnn1C1CC1)=O)=O CCC(C(=O)N1CCC(CCC(=O)NCCN(C)C2CC2)CC1)C(F)(F)F Cc1cc(N)c(C(=O)NCC2(C(C)NC(=O)CO)CC2)cc1F c1(NC(c2ccc(NC(C(C)OC)=O)cn2)=O)cc(COC)ccc1Br CCCCC(O)CC(=O)NCc1csc(CNC(=O)C(c2ccccc2F)C)n1 c1(CN(C(=O)CCCn2cc(-c3cnn(C)c3Cl)nn2)CC)ccccc1OCC C1(CNS(=O)(=O)C(F)(F)F)CCN(c2ncncc2F)CC1O c1(C(=O)NC2CC(NC(c3c(COC)noc3)=O)C2)cc(N)ccc1F Cc1c2c(nn1C)CCC(NC(=O)CCCCCn1cc(C3CCCO3)nn1)C2 N1(C(C(c2ccc(Cl)cc2)OC)=O)CCCC(O)(CNC(=O)C(C)(C)F)C1 C(=O)(CC1c2ccccc2C(=O)N1C)NC1(C)CC(NC(CC(C)C(F)F)=O)C1 c1(-c2ccc(C3CCN(c4nccc(OC)n4)CC3)o2)ccc(Cl)c(Cl)c1 S(=O)(=O)(c1ccc2c(c1)CCO2)NC1C(C(=O)NC2CCNCC2F)CCCC1 N1(C(CCOC)=O)CCC(O)C(C)(C)C1.C1(N2CCCC2=O)CC(C)C2CC12 N1(Cc2c(C(=O)O)cccc2)Cc2[nH][nH]c(=NC(=O)C(F)(F)Cl)c2C1 C(=O)(CCC(C)CN(C)C)N1CCC(CCNC(C(COCC)(C)C)=O)C1 C12(CC(=O)Nc3ccc(C)nn3)CCCC1N(C(=O)C=CCN1CCCC1)CC2 c1(OCC(=O)NCCCCCNC(c2cc(CC)ncc2)=O)cccc(C#N)c1 Cc1c(C(=O)NC2CC(NC(c3ccn4ncnc4c3)=O)C2)c[nH]c2nccc1-2 C1(NC(c2cc(SC)oc2)=O)CCCC2CN(C(c3ccc(C)c(O)n3)=O)CC12 c1(CC)cccc(C(=O)NC2CCCCC2NC(C2(C)CC=CCC2)=O)n1 C12(C(=O)NCCSCCC=C)CC1CCN2C(=O)C(C)S.C(C)(C)N N(C1CCC(C)(C)c2ccccc21)C(c1c(OC)ccc(S(=O)(=O)F)c1)=O C(CCC(C)C(=O)N1CCOC(CNC(=O)CCc2cc(C)cc(C)c2)C1)OC CN1C(=O)NCC1C(=O)NC1CCN(C(C2CN(C3CCCCC3)C2)=O)CC1 c1(CC)cc(C(N2CC(O)(CCNC(=O)Cc3ccccn3)C2)=O)nn1CCO c1(C(N2C(C(=O)NCCCCC#C)CC3CC32)=O)ccc(Cl)c(C#N)n1 C12(NC(CC3(NC(C)=O)CC3)=O)COC(C1)C(NC(c1snnc1C)=O)C2 C1(C(N2CC(C(=O)NCCc3cn(C)cn3)(COC)C2)=O)CCCCC1(C)C N1(CCCSc2ccccc2)CCC(C2CCCNC2)C1 CCC(CC)C(=O)NC1CCC(C(=O)NC(c2ccc(C)nc2)C)C1 c1(CN2CC3(CC(C(=O)NC4(C(=O)OC)CCC4)C3)C2)cccc([N+](=O)[O-])c1Br CN1CCC(c2nc(CCCCF)n(-c3ccccc3)n2)CC1 C(C(C)(O)C(=O)NCC1CCCN(C(C2CN(C3CCOC3)C2)=O)C1)OC c1(CC(=O)NCC(CNC(Cc2cc(C)no2)=O)F)c(C)cccc1F c1(C(CO)NCc2ncccc2Br)cccc(C(F)(F)F)c1 Cc1cc(=NCCCn2nc(C)c(CCNC(=O)CN(C)C)c2C)[nH]cc1F C1(C(=O)NC2CCC(F)CC2)(CNC(C(SC)SC)=O)CC2(CC2)C1 CCC(CC)(CCNC(C1CCCC1)=O)NC(c1cc(C(C)(F)F)on1)=O CC(C)CCC(c1nnnn1C)NC(c1ccc(C(C)(C)C)cc1)C c1(CC)ccc(C(=O)NCC2CC(NC(=O)Cc3ccnn3C)C2(C)C)cc1Cl c1(CC)cccc(C(N2CC(CNC(=O)C(=O)Nc3ccccc3)CC2C)=O)n1 N1(C(CC=CC=C)=O)CC2(CCCC2)C1C(=O)NC(c1cnccn1)C N1(C(C=C(C)Cl)=O)CC(NC(c2ccc3cccnn23)=O)CC(C)(C)C1 N1(C(C#C)(C)C)CCN(C(=O)C(=O)NCc2cccnc2Br)CC1 C=CCCCC(=O)NC(C1CN(C(=O)C(c2ccc(Cl)nc2)(C)C)CCO1)C C(=O)(CC(C)C(C)(C)C)NCc1occ(C(N2CCC(C(C)C)C2)=O)n1 n1(CCC(=O)N(C)CC2CCN(C(=O)CCc3cnn(C)n3)C2)cnccc1=O N1(C(=O)C2=CCCCC2)CC(NC(C2CC(CC3CC3)C2)=O)C2CCCCC12 Cc1cc(Cl)c(C(=O)NCCC2CC(NC(=O)C(C)Cn3ccnc3)C2)cc1N C1(COC)CN(C(=O)C(c2ccccc2)=O)CCN1C(c1cccnn1)=O O=C1Cc2c(N(C3CC(N)C3)C(=O)Cc3cccc(O)c3)ncnc2N1 CCCC(C(=O)NC1(C)CC(NC(=O)C(=O)NCC)C1)S(N)(=O)=O CCCCCC(CC)C(=O)NC1(C2CCCN2c2cc(C(N)=O)nc(Cl)n2)CC1 c1(C(N(CC(CN(C(C(=O)NC(=O)NCC)C)C)O)C)=O)ccc(Br)nc1N c1(C(=O)NCCCC(C)NC(=O)C(c2ccc(F)cc2)(C)C)cc(Cl)nn1C c1(C(=O)NC(C)C(N2CC(=O)NCC2CN(C)C)=O)cc[nH]c2nccc1-2 C1(CC(C)C)C(=O)N1.C1(CCN(C)C)C(=O)N1.C(C)(C(=O)N(C)C)OC c1(CCOC)ccc(NC(=O)CC2(C)CCN(C(=O)COCP(C)(C)=O)C2)cc1 C(=O)(C1COc2ccc(F)cc21)NCC1(F)CN(C(C(P(C)(C)=O)O)=O)C1 C(C(C)(C)CCNC(C1(C)CC1Br)=O)NC(CCOCC(C)C)=O C(=O)(C1CCCc2cncn21)NCC1=CCN(C(C=CC(=O)OCC)=O)CC1 C(CS(=O)(=O)NCCCCN=[N+]=[N-])(C1CCCCC1)OC C1(NCc2cnc(CCC)s2)CCC(C(=O)NCc2nc(Cl)sc2Cl)CC1 c1(C(N2CCC(C)SCC2)C(=O)NC2CCC2)ccc(F)c(Cl)c1F C(C(=O)NC(CC(=O)N1CCCC1CC1CCC1)C1CC1)(C(C)C)OCC N1(C(CCCc2cc(C)sc2C)=O)CC(C)(C(=O)C(=O)O)CC1(C)C C1(C(N2CC(NC(C3CCC4(CCC4)C3)=O)(CO)C2)=O)CCc2ncccc2C1 c1(CC(=O)NCCC2(C(N3CC(C)(OCC)C3)=O)CCC2)cnccc1C Cc1ccc2c(c1)SC(C(N1CC(CN(C)C(C3CC4(C3)CC4F)=O)C1)=O)C2 N1(C(c2onc(C)n2)C(=O)Nc2ccccc2Cl)CCc2[nH]nc(CO)c2C1 C1(CCNC(c2c(C)onc2)=O)CSCCN1C(c1cccc(O)c1)=O c1(CC(N2CCN(CC(=O)NC(C)CCO)CC2)=O)c(F)cc([N+](=O)[O-])cc1F C12(CNC(C(C)c3ccon3)=O)CC1CN(C(=O)CCN1CCC1)C2 N1(C(c2cccc(OCC)c2N)=O)CCCC2(CCC(NC(C)=O)C2)C1 N1(C(C2C(=C)C2)=O)CC2CCC1CC2NC(=O)C=C(C)C(C)(C)C N1(C(c2c(OC)ccc(F)c2)=O)CCC2(CCN(S(=O)(=O)c3cccc(C)c3)C2)C1 C(CCN=[N+]=[N-])CN(CCCC1(C(=O)OCC)CC1)C.C1(=O)CO1 c1(CC)nc(C(=O)NC(CC2CC2)C(N2CCC(O)(C(N)=O)C2)=O)c(C)o1 CC1C(C)N(C(c2cc(C#N)ccc2N)=O)CCN1C(c1cncs1)=O c1(SC)cccc(C(=O)NCC2(C)CN(C(=O)CS(=O)(=O)N(C)C)CCO2)c1Cl C1(CNC(=O)Nc2c(OCCC)cccc2)CC2(CCC2)C(=O)O1 c1(C(N(CCNC(=O)CCCN2CCCC2)CC2CC2)=O)ccc(Cl)cc1 c1(CNC)ccc(NC2CCCN(CC(=O)OC)CC2)cc1C#N c1(C(CNC2C(CC(C)C)C2)NC(=O)C=C(Cl)Cl)ccc(N2CCCCC2)cc1 C1(CNC(CC(CC=C)(C)C)=O)CCN(C(c2cnns2)=O)CCC1(F)F CC1(C)CC(NC(c2cccc(N)n2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C1 C1(CNC(CN(CC(C)C)C(c2ccccc2)C)=O)Cc2cccc(F)c2O1 N1(C(N)=O)CCN(C(C2COCC2NC(=O)C=CC(F)F)=O)CC1 C1(CC(=O)NC2(CNC(C3(C)C=CCCC3)=O)CCCCC2)CCCC(C#N)C1 C1(NC(NC(CC=C)C)=NCCC(=O)N(C)C)CCC(C)c2ccccc2C1 CN1CCC2(CC1)CN(C(C1(C3CC3)CN(C(C3CCC(F)CC3)=O)C1)=O)C2 Cc1[nH]c(C(N2CCC3(CCSC3)C2)=O)c(C)c1C=O C1(C)(CNC(C(COCC)n2cc(C3(C)CC3)nn2)=O)CC=CCC1 c1(C(C)NC(c2sccc2I)c2nnnn2CCCF)cccc([N+](=O)[O-])c1 c1(C)noc(CC)n1.C(=O)(CC(C)n1ccnc1)N(N(CC(CN(C(C)C)C)O)C)C Nc1cc(Cl)c(Cl)cc1C(=O)NCCC1CCN(C(C2OC3CCC2CC3)=O)C1 C1(C(N2CCC(C#N)C2)=O)CC2CC1CN(C(c1coc(N(C)C)n1)=O)C2 CC1(C)CCCC(C)(NC(C2CCC3(CC3)N2C(=O)CC2=CCCC2)=O)C1 C(=O)(C1CCCc2ccnn21)N1CCN(CCNC(c2c(C)nc(O)[nH]2)=O)CC1 C1(C(N(CCNC(C(C=C)(C)C)=O)CC)=O)CCCC(C)CC1 C1(C(=O)NC2(CNC(C3CC(C#C)(O)C3)=O)CC2)CC1C1CCCC1 CC1(C)CC(NC(C2CC(CNC(=O)CC3CCC4CC34)C2)=O)C1 CCCCN=C(NCCC1CC1)NCCF.c1(CCC(=O)N)ccccc1C N1(C(COC2CN(C(C)=O)C2)=O)CC2(C)CN(C(=O)C(CO)N(C)C)CC2(C)C1 C(CCCCCC(=O)NCC1CCC(C)(C)O1)NC(C(CC)COC)=O c1(C2(CNC(=O)NC3CC3)CC2)cc(F)ccc1F.N12CCCC(C1)NC(=O)C2=O Cc1cc(C)c2c(c1)C(N(C)C(=O)Cc1ccc3c(c1O)OC(F)(F)O3)CCO2 C12(NC(C3CC(OC)C3)=O)CC(CO)(C1)OC21CN(C(=O)CC2CCCCO2)C1 N1(C(c2c(Cl)cn(CCC)n2)=O)CCC(O)C(NC(c2nc(C)oc2C)=O)C1 N1(C(CCCNC(C)=O)=O)CCOC(CCCNC(C2CC3CC3C2)=O)C1 N1(C(C(C)(C)N(C)C)=O)CC2CCC2(CC(N2CC3CC2CN3C2CC2)=O)C1 S(=O)(=O)(c1ccc(Br)s1)NCC(=O)OC.C1(=O)C(C)(OCc2ccccc2)CCO1 C1(C(=O)NCC2CC(F)(CNC(CS(=O)(=O)NC)=O)C2)CCc2cnn(C)c2C1 c1(N2CCN(C(c3c(OC)ccc(OC)c3)=O)CC2)cc2c(cn1)C(=O)CCC2 c1(CC(=O)NCC23C(CN(C(C(CC)O)=O)C2)C3)ccc(C)c(Br)c1 C(=O)(NNC(=O)c1cc(C#N)on1)c1cn(CC(C)C2CC2)nn1 c1(C(=O)NCC(C(C)C)NC(c2cn(C)nn2)=O)ccc(Br)c2cccnc12 c1(OC)ccc2[nH]cc(C(N3CCN(Cc4cnc(F)cc4C)C4CC34)=O)c2n1 C(CC(=O)NCc1nc(C(N2CC(O)(C(C)C)C2)=O)co1)(c1ccccc1)OC c1(SC)ccc(NCC(N2CCCC2CNC(c2cccn2C2CC2)=O)=O)cc1 c1(C(=O)NCCN(C(c2ccc(F)c(C(F)(F)F)c2)=O)CC)cc(F)c(F)cc1O N1(C(C(C)C2(O)CCC2)=O)CCC2(CCN(C(C3(NC(N)=O)CC3)=O)C2)C1 O=C(C1=CCCOCC1)NCCC1CCCN(C(=O)COC(F)(F)F)C1 Cc1cc(C)c(OC(c2ccccc2)C(=O)NC2CCC(C)C2)c(C)c1 C1(NC(CC(=O)OC)=O)CN(C(C2CCCN2C(C)=O)=O)CCC1(F)F C1(NC(CN2CC(NC(CN(CC(=O)NC(C)C)C)=O)C2)=O)CCCC(CO)C1 c1(C(N2CCC(C(CC)CC)C2)=O)ccc(N2CCN(C(=O)NCC)CC2)nc1 N1(C(c2cncc(N(C)C)c2)=O)CC(CNC(=O)Cc2cscc2F)C2(CC2)C1 CCC(C)CCCC(=O)NCC12CCC(CC1)N2C(C1(N=[N+]=[N-])CC1)=O C1(NC(=O)CC2CC2)CN(C(c2nc[nH]c3nccc2-3)=O)C2(CCCC2)C1 c1(NC(CC(C)NC(C2CCC(NC(C)=O)CC2)=O)C)nnccc1C#N c1(NC(c2n(CC)ncn2)=O)cccc(NC(=O)CCC2CC(C)(C)CO2)c1 n1(C(CC)C)nnnc1C(C)(CCN1CCSCC1)NCc1ccoc1C N1(C(CP(C)(C)=O)=O)CCOC2(CCN(C(=O)C3=C(Cl)CCCC3)C2)C1 Cn1nnc2c1C(C(=O)N1CC3C(C(N4CC(S(C)(=N)=O)C4)=O)C3C1)CCC2 C(=O)(CC(C)CCC=C(C)C)N1CC(COC)N(C(=O)CC2CC3(CC3)C2)CC1 c1(C(=O)NC2C(CNC(c3cn(CC)nn3)=O)CCC2)c(C)ccc(Cl)c1F C1(C(C)O)CCC(NC(c2cccc(CO)n2)=O)CC1.C12(C(=O)N)CSCC1C2 C1(C(N2C(CCNC(CCSCC(N)=O)=O)CSCC2)=O)CCCCC12CCC2 c1(C(=O)OC)cc(C(=O)NC2CN(NC(C)=O)C2)ccc1C.C12CC1C(=O)N2 c1(C(=O)NCCOC(CNC(CC(C)C2CC2)=O)(C)C)nc2ncccn2n1 C1(Nc2ccccc2)CN(c2cc(NC3C(C(=O)OC)C3)ncn2)CC1OC C1(C(C)NC(c2n(CC)ccc2)=O)CN(C(c2cnncc2C)=O)CCO1 C1(C(=O)N(CCCC(=O)OC)C)(OC)CCN(C(=O)C(c2ccc(C)cc2)F)C1 c1(CCC(=O)NCC2C(NC(C3(C#C)CCC3)=O)COC2)ccc(SCC)cc1 c1(C(=O)NC2(C(N3CCC(C#N)CC3)=O)CCCC2)cccc2c(Br)n[nH]c12 C(=O)(C(C)(CNC(C12CCC(C1)C2)=O)CC)N(C(C=C)C)C Cc1ccc(NCC(=O)N(C)CC2CCCN(C(=O)C=Cc3cscn3)C2)cc1 C1(c2onc(CC3CC(C)(CO)C3)n2)CCCCC12CC2(F)F C1(CNC(CCc2scc(C)n2)=O)C2CCCC1N(C(=O)CCC1CCCC1)C2 C1(NC(C2CC2F)=O)CCC(NC(c2csc(Cc3ccccc3)n2)=O)CC1 CC(C)(O)C(F)C(=O)NC1(C2CN(C(c3cc(-c4cccs4)[nH]n3)=O)C2)CC1 N1(C(C2(OCC)CC2)=O)CC2OC(=O)N(c3ccccc3)C2C1.C1C=CC(=O)N1 C1(C(=O)NC2CC(CC(=O)NC(C3CCC3)C)C2)CCC(N2CCCC2=O)CC1 C(=O)(C1Cc2cccc(Br)c21)N(C)CC1CC(C(=O)OC)C1 C1(CCNC(c2coc(CNC(C3(O)CCCCC3)=O)c2)=O)CC2(CCO1)CC2 C1(C(N(C2CCN(C)CC2)C)=O)CCN(C(=O)CC2CCCC(=O)C2)CCO1 N1(C(C(CC#C)C2CC2)=O)CCC(O)C(F)C1.C1(C(=O)NCC)CCC1 C(=O)(CCC(=O)N1CCCCC1c1n[nH]cc1C(=O)NC12CC(C1)C2)NC c1(C(=O)NC2C(NC(c3cnc(CCCC)[nH]3)=O)CCCC2)ccc(C)cc1Cl C(CC)(C(=O)NCC1CCC(NC(=O)C(CC)OCC2CC2)C1)=CCCC c1(OC)c(C(N2CCC(C)(NC(=O)CN(C)C(C)C)C2)=O)cc(Cl)cc1Cl c1(C(N2CCC(O)(CNC(C(CC)NC(N)=O)=O)C2)=O)cc(C)ccc1Cl Cn1ncc2c(C(=O)N(C3(CO)CCOC3)CCO)ccnc12 N1(C(C(C2CCCCO2)N)=O)CCSC(C(F)(F)F)CC1 c1(NC(C2CN(C(C3CCC(C)O3)=O)CC(F)C2)=O)ncc(Br)cc1[N+](=O)[O-] C12(NC(c3cc(OC)c(F)cc3N)=O)CCC(CN(C(=O)Cc3cscn3)C1)C2 O=S(=O)(c1ccc(NCC2CC(CO)CO2)c(F)c1)NCc1cc(O)ncn1 C(CCCCC(=O)NCC(CNC(C1COC(=O)N1C)=O)C(F)(F)F)N(C)C C1(C(=O)NCC(=C)CCNC(c2cnnc(C)c2)=O)CC(O)CC(C)O1 c1(C(=O)NC2CN(C(c3cc(C)sn3)=O)CC(F)C2)cc(C)c(F)cc1F C1(NC(CN(C)C)=O)CC2CC1N(C(=O)Cc1sc(O)nc1O)C2 Cc1[nH]cc(C(N2CC=CC2CNC(c2cnn(C)c2C)=O)=O)c(=O)c1Cl C1(C(=O)NC2CN(C(C3(CC(C)C)CCC3)=O)CC23CC3)CC2CCC(C1)C2=O C=C(Cl)C(C)(C)C(=O)NCC1(NC(c2cc(CO)c(C)o2)=O)CCOC1 c1(OC)cc(F)c(C(=O)NCC2C3CN(C(c4ccncc4N)=O)CC23)cc1N CC(CCCNC(=O)C(C)c1cc[nH]n1)NC(C1OCCO1)=O N1(C(C(CCC)OCC)=O)CC(=O)NCC1C(=O)NOCCO C1(CNC(CNC(=O)OCC)=O)CCCCC1NC(C1CC(F)CN1C)=O C(CC(CNC(=O)C(C)Cc1ccccc1)NC(c1cc(C)no1)=O)OC S(=O)(=O)(c1ccc(NC2CCC2O)c(Cl)c1)NCc1c(F)ccc(C)c1 C(=O)(C1=CCC(C)CC1)N(C)CC1N(C(C(C=C)C)=O)CCC1 C1(C(=O)NC2(COC)CN(C(C3(C)CCCS3)=O)C2)CCc2nnnn2C1 C(=O)(C1CCc2cc(F)ccc21)NC1(COC)CCN(C(C2COC(=O)N2)=O)C1 C1(C2CN(C(=O)C(c3cccc(O)c3)C)C2)(NC(Cn2ncc(C)c2)=O)CC1 C1(C(=O)NCC(CCCCC)O)CN(C(=O)CCC(C)(C)OC)CC(C)(C)C1 c12ccc(NC)c(c1)OC2=O.C1(CNC(COC)=O)CCN(C(C2(CO)CC2)=O)C1 N1(C(C(N2CCOC2=O)C)=O)CCOC(C(N2CC(n3ccnc3)C2)=O)C1 N1(C(COCC)=O)CCCCC1C1CCCN1C(=O)Cc1nc(C)cs1 C1(O)(CNC(c2c(CC)ocn2)=O)CCN(C(c2c(C)[nH]c(CC)c2C)=O)CC1 n1(CC(=O)NC2CCN(C(C(C)C#N)=O)C2C(C)(C)C)cc2ncccc2n1 c1(C(N2CCOC(CO)C2)=O)cc2cc(-c3cnn4ccccc34)ccn2n1 C1(CNC(C(C(C)C)n2ncc(C)c2)=O)CN(C(=O)CC2CSC2)CC1(F)F C(=O)(C(C)CCC(C)(C)C)N1CC(CN(C(=O)COc2ccsc2)C)OCC1 c1(CCC(=O)NCC(C(=O)N(CC(C)NN(C)C)C)N(C)C)cccnc1F.CC C1(C(=O)NCCCCCN(C)C)CN(C(=O)CCc2ccn(C)n2)C2(CCC2)C1 c1(CC)cc(C)c(C(=O)NC2CC3(C2)CC3NC(c2ccc(C(F)F)cn2)=O)o1 C1(NC(CSC)=O)CCN(CCNC(C2CC2c2ccco2)=O)CC(C)(C)C1 C1(C(C)NC(=O)C=Cc2cccs2)CN(C(=O)CC=CC(C)(C)C)CCO1 C(=O)(CCCCCCNC(=O)CC1CC(C(N)=O)C1)N(CCC(=O)NC)CC CC1CC(NC(c2ccc(C3CC3)cc2)=O)CN(C(c2cc(F)ccc2O)=O)C1 c1(C(N2CCCCC2C)C(=O)NC(C)C)ccc2c(c1)CC(C)(C)O2 N1(C(c2cn(C)c(=O)cc2)=O)CC2CCCN(C(=O)CC3CC3)C2C1 c1(C(=O)NCC(CNC(CNS(N)(=O)=O)=O)F)ccnc2ccc(N)cc12 CC1(C)CC(C)(C(=O)NCC(C2CCCC2)NC(c2ccn(C3CC3)n2)=O)C1 c1(C(N2C(CNC(=O)Cc3cncs3)CC2)=O)cc(-c2ccccc2)ccc1N Cc1ccc2c(C(=O)NC3COCC3NC(C3CCOC(C)(C)C3)=O)coc2c1 C1(C(=O)NC(CC(C)NC(C2CC(=C3CCC3)C2)=O)C)CCCC2(CC2)C1 C1(C(=O)NCC2N(C(CCNC(=O)CO)=O)CC(O)C2)CCCC1C1CC1 N1(C(N2C(C=CC)(NC(=O)CCCCC(C)C)CC2)=O)C2CCC1CC(OC)C2 CN1CCC(C(=O)NCC2(CC(=O)NCc3ccc(O)cc3F)CC2)CC1=O c1(C(=O)NC23CC(C2)N(C(C2CC2C2CC2)=O)C3)cc2c(cc1Cl)OCCO2 C1(CNC(C(C(C)C)(C)C)=O)CN(C(=O)CCCCC2CC2)C2CCN1C2 C(=O)(C(C(C)C)n1cccc1)NC(C1N(C(c2n(CCC)ncc2)=O)CCC1)C N1(C(CC(C=C)CCC)=O)Cc2ccccc2C(NC(=O)CN2CC3CC3C2)C1 c1(C(=O)NCCN(C(C(C(C)OC)O)=O)C2CC2)cc2c(cn1)CCCC2 c1(OC)cc(CC(N2CCC(C)C(NC(=O)C(F)=C(C)C3CC3)C2)=O)ccc1C O=C1NCCCCC1C(N1CCC(CNC(=O)C(F)(F)C(F)F)C1)=O N1(C(C2CC(OCC)C2)C(=O)NCC)CCCC(C)(C(C)C)C1 C1(COCC(=O)NCC(F)F)CN(C(=O)COCCc2ccco2)CCO1 Cc1c(C(=O)Nc2ccc(NC(C3(CO)COC3)=O)cc2)cccc1C1CC1 Cc1c(C(=O)NC2CCN(C(C3(CS(C)(=O)=O)CC3)C)C2)oc2c(C)cccc12 C1(C(=O)NC(C(C)C)CNC(c2cc(C(C)(C)C)no2)=O)CCC(C)CC1 CC1(C)CN(C(c2csc(S)n2)=O)CC1NC(=O)CCC1CCCCCC1 N1(C(c2c(C)n[nH]c2C)=O)CC(NC(c2ccc(Cl)cc2)=O)CC(O)C1 C1(NC(CC2CCC(C)CO2)=O)C2CC3C(C2)C13CO.C12(C)CC(C1)C(=O)N2 n1(C(C)(C)C)nc(C(N2CCN(C(=O)CNC(C3CCC3)=O)CC2)=O)c(Br)n1 C1(CN(C(C2SC3C=CC2C3)=O)CC)CCN(C(=O)C=C(C)COC)CC1 CC1C(NC(=O)CN2CC(=O)N(C)C2=O)CC2CCC1N2C(=O)C=C(Cl)Cl c1(NC(C)CCNC(=O)Cn2nnc(=N)[nH]2)cc(=O)n(C)c(=O)n1C c1(C(=O)NC2C(CNC(=O)Cc3csc(=N)[nH]3)C2)cccc(OCCBr)c1Cl C(=O)(C1CCCc2c[nH]nc21)N1C2C(NC(c3cncc(Br)c3)=O)C(C2)C1 c1(OC)cc(C(N2CCC(CCNC(=O)CC3C=CCC3)C2)=O)ccc1[N+](=O)[O-] Cc1cc(-c2nc(Cc3cccs3)nn2-c2cnnn2C)c2ccccc2n1 Cc1ccc(NC(=O)CC(C)NC(C2CC3CC3C2)=O)cc1[N+](=O)[O-] C1(CC(=O)NCC2(F)CC(CNC(c3ccsn3)=O)C2)(COC)CCCC1 C1(C)(CC)CCCN(C(=O)C2=CCN(C(=O)Cc3csc(C)n3)C2)CC1 c1(C(=O)NCC(CCCC)NC(C2(Cl)CC2(C)C)=O)cc(C)c2nc(C)cn2c1 N1(C(COCC(C)C)=O)CC(CC(=O)NC2C=CCCC2)CC1(C)C CC1CC(NCc2ccc(C#N)cc2)CC(C)(C)C1 N1(C(C2N(C(CC)=O)CSC2)=O)CC(CN(C(=O)C(F)(F)CC)CC)C(C)C1 Cc1cc(Cl)cc(Br)c1NC(c1nc(C(=O)NCc2c(F)cccc2F)cs1)=O c1(C2(C(=O)NCC=CCNC(c3nnn(C)n3)=O)C(C)C2)c(Cl)cccc1Cl Cc1nccnc1C(=O)NCC1CCC1NC(=O)CS(N)(=O)=O c1(C(C(=O)NCCCCCCNC(=O)C=CC2CC2)O)ccc(Cl)cc1Cl CS(=O)(=O)c1cnc2c(-c3nc(-c4ccc5sc(C(=O)O)nc5c4)no3)cnn2c1 C1(NC(C(C)N2CCC2)=O)CC(F)CN(C(c2ccc(C(F)(F)F)cc2Cl)=O)C1 c1(N2CCC(C(C)NC(=O)CC3CCCOC3)CC2)ccc(C#N)cc1[N+](=O)[O-] C1(NC(c2cn(C3CC3)nn2)=O)CCN(CCF)CC1.C123CC(C1)(C2)CNC3=O C1(NC(C(CC)(C)CO)=O)CC2CCC1CC2NC(=O)CC1CNC(=O)O1 N1(C(C2(CNC(=O)CCNC(=O)CO)CC(=C)C2)=O)CCC12CCCSC2 N1(C(C=C(CC)C)=O)CCC(NC(=O)CCOCCOC2CCCO2)CC(O)C1 C(C(=O)NC1CN(C(=O)C(F)(F)CO)CC1F)(c1ccccc1)=CC(C)(C)C N1(C(C)=O)CCOC(C(=O)NCC(C2CCSC2)NCc2ncccc2O)C1 Cc1nc(C(=O)NC2(CNC(c3ncc(Cl)cc3F)=O)CCC2)cn(C)c1=O N1(CCOC)CC(C(N2CCOC(CNC(C3(O)CCCCC3)=O)C2)=O)CC1=O C(c1ccnn1C)=CC(=O)NCC(CC=C)NC(=O)C(O)CCN(C)C c1(N2CC(CNC(=O)CCc3cccnc3)OCCC2)ncnc2cnccc12 c1(NC(C(C)(N(C)C(C2CCC=CCCC2)=O)C2CC2)=O)ccc2c(c1)OCO2 CCCCC(C(=O)NCc1ncc(C)cn1)NC(=O)CC1CCC(=O)N1C N1(C(c2ccc(OC)c(O)c2)=O)CCC2C1CCCN2Cc1cc(Br)ccc1I c1(C(N2CC(NC(C3C(C=C)C3)=O)C2)=O)cn(C)nc1-c1ccco1 C(C(CC(=O)NC1(CNC(c2ccnnc2S)=O)CCCC1)C(F)(F)F)N(C)C C(C(CC(F)(F)F)NC(c1ccc(OC)s1)=O)NC(c1cc(CC)on1)=O c1(C(N2CCOC(c3nc[nH]n3)C2)C(=O)NCC=C)cccc2[nH]ncc12 C12CCC(CC1)NC(=O)c1nccc(n1)CC(=O)N2C.CC1CCCC1C(N)=O N1(C(c2c(CCC)c(C(C)=O)c(C)[nH]2)=O)CCOC2CCN(C(=O)C(C)O)CC12 c1(CC)ccc(C)c(C(=O)N(CCNC(=O)CCCn2cc(C)cn2)C2CC2)c1 C1(CC(=O)NC(COC)CNC(c2cc(C3(C)CC3)on2)=O)CCC(=O)NC1 C1(C(=O)NCC2(C)N(C(CCC3(C)CC3)=O)CCC2)C2CCC(C2)C1(C)C c1(C(=O)NC2CC(NC(C3CC(OCC)C3)=O)C2)cc2cc(Cl)ccc2o1 CCCC(C(O)C(=O)N(C(C)C(=O)NCC)C)NC(c1ccccc1CC)=O CCC(C)C(O)C(C)C(=O)N1CC(C(=O)NC2CCOC2(C)C)C1 Cc1coc(C(C)C)c1C(N1CCC(C)(CNC(c2csc(C(F)F)n2)=O)C1)=O C(=O)(C1=CCCN(C(=O)CC(C)C2CCCC2)C1)N1CCC(OCC)CC1 C(=O)(C1=CCN(C(c2ncnc(O)c2F)=O)CC1)NCC(c1nccs1)C N1(C(CCc2onc(C)n2)=O)CCC(F)(CNC(c2sc(O)nc2C)=O)C1 c1(N2CC(CC)OCC2)nc2c(c(=NCC3CC4C(C3)C4(F)F)[nH]1)CCCC2 N1(C(c2c(C3C(C)C3)nccc2)=O)CCCC(n2cc(-c3cc[nH]n3)nn2)CC1 C1(OC)CCN(C(=O)CCC2CCC(NC(=O)COCCCF)C2)C1(C)C N12CCC(CC1)CCN(C)CC2=O.C1(NC(C=C(CCC)C)=O)CCC(C)O1 c1(OC)ccc(C(=O)N(C2CN(C(=O)CCc3nc(C)no3)C2)C)c(F)n1 CCCC(CC)CC(=O)NC1CC(NC(=O)C(c2ccccc2Cl)(C)C)CC1O c1(OC)c(Cl)nc[nH]c1=NCC1CC(NC(c2cnc(N(C)C)c(Cl)c2)=O)C1 c1(C(=O)NCC2C(NC(Cn3nnc(C)n3)=O)CC2)cc(F)c(F)c(Cl)c1F N1(C(C=C2CCC(C)C2)=O)CCC2(CCCN2C(=O)CCC(=O)N(C)C)CC1 N1(c2cc(N3CC(c4n(C)cnn4)C3)ncn2)CCC(C2CCCCC2)CC1 c1(C(N2C(CCNC(c3conc3C(F)(F)F)=O)CCC2)=O)n[nH]c2c1COC2 Cc1cccc(CC(=O)NCCC(C)N(C(=O)CC2CC3(CC3)CO2)C)c1F N1(C(c2cc(OC)no2)=O)CCOCC1CNC(c1sccc1Br)=O C(c1ccc2c(c1)OCO2)=CC(=O)N(C)CC1CCN(C(C(CCCC)O)=O)C1 N1(C(c2cccc(C)n2)=O)CCN(C(c2cnc(C)nc2C)=O)CC2(CC2)C1 Cc1c(C(=O)NCC23CC(NC(=O)COCC(C)C)(C2)C3)cccc1C(F)(F)F C(C)(CNC(=O)C=CCO)(CNC(=O)Cc1ccns1)OC Cc1ccc2cc(C(N3CC4CC3CC4NC(=O)Cn3cnnc3O)=O)[nH]c2c1 c1(CN(CC(F)F)C(c2cccc(Br)c2)=O)nc2c(o1)CCSC2 CC(C)C(N=c1nc(C2CC2)[nH]s1)C(C)CNC(C1CC(C)(C)C1)=O c1(C(=O)NCc2cn(CC(=C)CC)nn2)cccc2ccc(C(=O)OC)nc12 CC(C)CC(O)C(C)C(=O)N(CCCCNC(C1(C(F)(F)F)CC=CCO1)=O)C C(CCF)(C(=O)N1CC(F)(C#N)C1)NC(Cc1nc(C)oc1)=O Cc1nnc2n1CC(C(N1CCC3(C1)CN(C(C1CCC=CO1)=O)C3)=O)C2 N1(C(C2(C#C)CCCC2)=O)CCC(CNC(=O)COCC2CCOC2)C(F)(F)C1 CC1(C)CC(C(N2CCC2COC(N)=O)=O)CN1C(=O)CC1CC=CCC1 C1(C(NCP(OCC)(C)=O)=O)C2CC3C(C2NC(C2CC(C)CCO2)=O)C13 N1(C(c2c(CC)c(C)sc2)=O)CC2CCC(C1)N2C(=O)COC1CCCCC1C C1(CC)CCN(C(C2CC2(C)C(F)F)=O)C(C(=O)NC23CCC(C2)OC3C)C1 c1(C(=O)N(c2ccnc(Br)n2)Cc2ccccc2)ccncc1NC1CC1(F)F Cc1cn(C)nc1C(=O)NCCC1CN(C(=O)C(C2CCOCC2)F)CCO1 Cc1cc(Cl)cc(C(=O)NCc2cn(C3CN(C(=O)COCC4CC4)C3)nn2)c1C N1(C(CCOCC(C)C)=O)CCC(NC(=O)CC2NC(=O)CNC2=O)C1(C)C N1(C(C2(SC)CCC2)=O)CCC2(CCCC2CNC(=O)CC2CC2C)CC1 CC1=NNC(=O)C1CC(N1CC(NC(C2(NC(N)=O)CCC2)=O)C(C)C1)=O C1(C(N2CCCC(c3nc(C)c(C)[nH]3)C2)=O)CN2CCN1CC2C c1(C(N2CCC(O)C2)C(=O)NCC2CCOC2)ccc(Br)cn1 c1(C(N2CCN(C(C3(C)CCNC3=O)=O)CC2CO)=O)cc(Cl)cc2c1OCC2 C1(NC(c2c(CCC)[nH]cc2)=O)CCN(C(=O)COc2ccc(Cl)nc2)CC1C CC1C(NC(=O)CCOC2CC2)CCCN1C(c1cc(C2CC2)on1)=O Cc1ccc(C(=O)NC2CS(=O)(=O)CC2NC(c2cccc(C)c2C)=O)c(F)c1 Cc1noc(C)c1CCCn1cc(CN(O)C(C2CC3CCCC23)=O)nn1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2(CC1)CC2CNC(C1CC(=C2CCC2)C1)=O Cc1c(C(N2CC(CCn3cc(CO)nn3)C2)=O)nnn1CC1CCCCN1C N1(C(C(CC=C)OC)=O)CCC(NC(c2cnc(C(C)(C)C)nc2)=O)C(O)C1 C(CNC(=O)C(O)Cn1cncn1)(CC(=O)NC1CC(F)(F)C1)OC Cn1c(=O)c(N(CCC(C)(C)O)C)nc2ccccc12 C1(C(N(C)CC2CCN(C(=O)CN(S(C)(=O)=O)C)C2)=O)Cc2nncn2C1 CCCCC(C(=O)NCC(C1CC1)NC(c1cc(Cl)ccc1OC)=O)NC(N)=O c1(C(N2CCC(C(N(C)Cc3cc(CC)on3)=O)C2)=O)cc(C)c(C)nn1 N1(C(c2cccc(OCC(F)(F)F)c2)=O)CCN(C(=O)CC(F)F)C(C(F)F)C1 C1(O)(CNC(Cc2cccc(OC(C)C)c2)=O)CCCN(C(C2(C)COC2)=O)C1 c1(OC)c(F)ccc(F)c1CN1CCC(NC(=O)CCc2cc[nH]n2)C(O)C1 Cc1ncc(C=CC(=O)NC2CN(C(=O)CC3CCN(C)C3=O)C2)c(O)n1 C(=O)(C1CCCc2n[nH]cc21)N1CC(COC)(CNC(c2cccc(SC)c2)=O)C1 N1(C(C2N(C(c3nc(C(C)C)oc3)=O)CC=C2)=O)CCC2CC1C(=O)O2 C1(CNC(c2c(C)onc2)=O)CC2CCC1N(C(=O)C(C)C(C)(F)F)C2 C1(C(N2CC(O)(CCNC(=O)COCCO)C2)=O)CC2CCC1O2 N1(C(c2ccc(CC)[nH]2)=O)CCN(C(c2cc(-c3ccco3)no2)=O)CCC1C N1(C(C(C(=O)OC)C)=O)CCC(O)(C(N2CC(C)(O)C2)=O)CC1 Cc1c(C(=O)NC(CC(C)C)C(=O)NCC2(C3CCC3)CC2)cccc1C#N c1(NC(C2CCC3(C(C(=O)OC(C)(C)C)C3)C2)=O)ccc2oc(S)nc2c1 CC(C(=O)NC(c1nocc1C(=O)NCCc1ccccn1)C)C(C)(C)C C12(C(=O)NCC3(C(=O)NC4C(COC)CCC4)CCOC3)CCC(OC)(CC1)C2 C1(C(N2CC3CN(C(C=COCC)=O)CC3C2)=O)Cc2cc(Br)ccc2O1 C1(N(C(C=Cc2ncc(C)[nH]2)=O)C)CN(C(=O)CCC2CCC2)CC1(C)C O(NC(=O)C(CCF)NC(=O)C(F)CC(C)(C)C)CCOCC C1(OCC)CN(C(=O)CC2(O)CN(C)C2)CC1CNC(c1cnn(CCF)c1)=O N1(C(CC(CN(C)C)C(F)F)=O)CCC2CN(C(=O)C(C)(Cl)Cl)CC2C1 C1(N(C(CCN(CC)CC)=O)C)CCCC(NC(=O)C=Cc2ccncc2)C1 C1(NC(c2ccncc2O)=O)CC2CCC(C1)N2C(C1CCC2CC2C1)=O Clc1cc(NC(c2sccc2Cl)c2nnnn2C2CCCCC2)cc(Cl)c1 c1cc(=NC2CC3(CCCO3)C2)[nH]c(N2CCOC(c3n[nH]c(C4CC4)n3)C2)n1 C1(OC)CN(C)C(C)(C(N2CC(CNC(c3cn4c(n3)SCC4)=O)C2)=O)C1 CON(CCC(=O)NCCS(=O)C(C)(C)C)C(=O)C(F)C1(O)CCC1 C1(CNC(CC(C)OC)=O)CCCC2CN(C(c3ccc4cnoc4c3)=O)CC12 N1(C(C=CCCC(C)C)=O)CC2(C1)CN(C(C1CC(CC3CC3)C1)=O)C2 c1(C(=O)NCC2C(CNC(c3cnc(C(=O)OC)s3)=O)C2)cn(C)c(=O)nc1O C12(CC(O)C1)C(=O)N2.C1(CCNC(=O)CC2(SCCO)CC2)CCCO1 c1(OC)c(Cl)nc[nH]c1=NCC(C)(CO)NC(C12CC(CN1C1CC1)C2)=O c1(OC)cccc2c(N3CC4CC3C3CC43)cc(C)nc12 C1(O)(CNC(CN2CC(C)(C)C2)=O)CCCN(C(C23CC2COC3(C)C)=O)C1 N1(C(c2cnc(CC)o2)=O)CC(NC(=O)C=CC2CCOC2)C(C)C1 C1(NC(C(CCC)OC)=O)CN(C(=O)CSCCC(C)C)C2CCCCC12 N1(C(CCCNC=O)=O)CC(CO)C2(C1)CN(CC1CC1)C2.n1(C2(CO)CC2)cnnn1 c1(COC)ccc(C=CC(=O)NCC=CCNC(=O)C2CC2)s1.C1(N)(SC)CC1 C1(C(=O)NCc2[nH]nc(C(C)C)n2)CCN(C(=O)CN2CCOC2=O)O1 Cc1cc(Br)cc(C(N2CCC2CNC(c2cc3c([nH]2)CCCC3)=O)=O)c1C C1(CN(C(=O)CC2CC(n3ccnc3)C2)Cc2ccccc2)CC(F)(F)CO1 C1(C(=O)NC2(CC=C)CN(C(c3ncc(F)cc3N)=O)C2)COC2(CCC2)C1 C1(CNC(CSC(C)(C)C)=O)CCN(C(=O)CC2COCCO2)CC1(F)F C(N=c1[nH]c(N2CCC(OCCF)C2)nc(=N)[nH]1)Cc1ccc(CC)cc1 N1(C(CCOC(C)=O)=O)CCCC(F)(CNC(C2CCNC(=O)C2)=O)C1 C(=O)(C(F)(CNC(c1sncc1C)=O)C(C)C)N(C)Cc1ccc(CC)o1 Cc1ccc(S(=O)(=O)Nc2cncc(C(=O)Nc3cccnc3C)c2)c(F)c1 c1(C(=O)NC2C(C(=O)OC)COC2)ccc(NC(C2CC(=O)N(C)C2)=O)cn1 c1(C(=O)NC2C(CC(=O)NC(C)(C)CC3CCCC3)C(O)C2)ccc(F)cn1 c1(COC)n[nH]cc1C(=O)NC1CC1NC(C1(C)CC1(C)C)=O N1(C(CN(C)C(c2c[nH]nc2Br)=O)=O)CCN(C(C2CC2F)=O)CC1 N1(C(Cn2cc(C(C)=O)nn2)=O)CC2CC2(CNC(=O)C(C2CCOCC2)C)C1 C1(c2n(C(C)C)nnn2)(NCCNC(=O)OC(C)(C)C)CC2(C1)CC(C)(C#N)C2 C1(C(N2C3C(NC(c4nc(C)nc(O)c4)=O)C(C3)C2)=O)CC2CCC1NC2=O c1(C(N(C2CCN(C(C(C)c3cncs3)=O)C2)C)=O)cccc2cncn12 C1(NC(C(N2CCOC2=O)C)=O)CC=C(C(=O)NCc2cccc(O)n2)C1 C(=O)(CCCCCC#N)NC(CCOC)CNC(=O)C1CC1 C1(Cl)(C(=O)NCCc2ccc(CC(C)C)cc2)CC2CCC1O2 c1(C(=O)NC2CCN(C(CC3(OC)CCCC3)=O)C2C2CC2)cc(O)nc(O)c1 C=Cc1cnn(C)c1C(=O)NCC(CC(C)C)NC(c1ccnn1C(C)CC)=O c1(C2C(=O)NCCN2C)ccc(C)cc1Cl.CCCC=CCCOC CC1(NC(=O)C(=O)NCCCCCF)CCNC1 Cc1cc(C#N)ccc1C(N1CCCC1C(=O)NCCOC(=O)C1CC1)=O N1(C(CC2C(C(=O)OCC)C2)=O)CC2(CNC(=O)CCc3cnco3)CC1CO2 c1(C(N2CC3C(CNC(C4CCOC4)=O)(CC3)C2)=O)cc2cc(Cl)cnc2[nH]1 C1(CNC(c2ccc(Cl)cn2)=O)CCC2(CCN(S(=O)(=O)C(F)(F)F)CC2)CO1 CCCC(CC)CCC(=O)NCC1CCCCN1C(=O)C(=O)NCC(F)F N1(C(C2(CC=C)CCOC2)=O)CCC2(C1)CN(C(C13CC(F)C1C3)=O)C2 n1(CC(=O)NC2CCCC(CNC(=O)CC3CC3)C2)c(O)nc2ccccc12 c1(CNC(=O)CC2C=CS(=O)(=O)C2)cc(O)nc(CNC(c2cscn2)=O)n1 N1(C(CC2ON=C(C)C2)=O)CCC(OC2CC(NC(=O)Cc3cncs3)C2)CC1 N1(C(C(CCCNC(CCCC(C)(C)C)=O)O)=O)CC2(CCCCCC2)C1 CCC(C)(C)CC(=O)NC1CN(C(c2ccnn(C)c2=O)=O)CCC1CO CC1(C(N2CC3CC2C3C(=O)Nc2coc3c2CSC3)=O)Cc2ccccc2N1 NC1CN(C(=O)C(=O)Nc2ncoc2C(F)F)CC2(CCOCC2)C1 CCN(C1CCOC1)N1CCCC(CCn2ccnn2)C1 N1(C(CCN(CCC)C)=O)CCCC(N(C)C(C2CC3CC2CO3)=O)CC1 C1(NC(C(c2cc[nH]n2)OC)=O)(CNS(C)(=O)=O)CCOC1 CC1(C)CC(NC(C2CCCCC23CC3)=O)CN1C(=O)CSc1ccc(F)cc1 N1(C(c2nc(C)n(C)c2)=O)CCC(NC(c2ccco2)=O)C(CO)C1 c1(C(=O)OC)[nH]c(C)c(C(=O)NCCOCCN(C)C(C2CCC(C)C2)=O)c1C N1(C(c2ccn(C)n2)=O)CCCC(C(=O)NC2CCOC2)C1 C(=O)(C1=NNC(=O)CC1)NC1(CC=C)CCN(C(c2cc(C)c(C)cn2)=O)C1 C1(NC(=O)C(N2CCCC2)C2CC2)CC(O)CN(C(=O)Cc2cscn2)C1 C1(C(=O)NC)CC2CCC1N(C(=O)CC)C2.C(C(=O)O)NC(=O)NCO C1(NC(COC)=O)CC(F)CN(C(C23CCCC2C3(F)F)=O)C1 C12(NC(c3n(CC#C)ccc3)=O)CCC(CNC(C3CC34CCC4)=O)(C1)OC2 N1(C(C2(C)CCC(C)C2(C)C)=O)CC=C(C(=O)NCCCC(O)CO)CC1 c1(-c2nc(CC3CCN(C(=O)NC4CC4)C3)on2)ccc(F)c(F)c1 O=C(C1=C(Cl)CCOC1)NCC1CC(C(F)(F)F)CCN1C(=O)C#CC1CC1 O=C1CN(CCC2CC2(Br)Br)C2COCCN12 CC1(C(=O)NC2CC3(C2)CC(NC(C24CC(F)C2C4)=O)C3)CCCCNC1=O C1(C(C)C)CCC(CN2CCCCC2CNC(=O)OC(C)(C)C)C(=O)N1 C(C(CC(C)C)C(=O)NC1(CO)CC(F)C1)NC(Cc1cc(C)on1)=O C(=O)(CC(C)C(C)(C)NC(c1ccc(O)nn1)=O)NC(c1cnn[nH]1)C N1(C(C(=O)NCC)CC2(C(=O)OC)CC3(CCC3)C2)CCc2nnn(CC)c2C1 C1(NC(C2Cn3c(C)nnc3C2)=O)CC2CCC1CN(C(=O)CC1=CCCC1)C2 N1(C(C2(N=[N+]=[N-])CC2)=O)CCOC2CCN(C(=O)CN3CCCCCC3)CC12 C(CC(=O)N=c1ccn(CC2CC2)[nH]1)N(C(CCCOCCC)=O)CC c1(C(=O)NC(CN(C(C(C)Sc2ccc(C)cc2)=O)C)C)nc(Cl)ccc1Cl C(C(=O)N=c1ccn(C(F)F)[nH]1)C1N(C(C(CC)CC(C)C)=O)CC1 C1(CNC(C2(C)CC(=C)C2)=O)CCN(c2nc(C(C)C)cc(C)n2)CCC1(F)F CCCC(CC)C(=O)N1CCC(OCCNC(c2nccc(OC)c2F)=O)C1 C1(NC(COCC)=O)COC2(CCN(C(c3cc(Br)c(C#N)s3)=O)C2)C1 N(C1COc2c(Cl)cc(Cl)cc21)c1c2cnn(C(C)C)c2nc(Cl)n1 N1(C(C2CCN(C(N(C)C)=O)CC2)=O)CCCC2(NC(C3CC3(F)F)=O)CC2C1 c1(C(C(=O)NCCC(=O)OC)N(CC(=O)NCc2cccs2)C)ccc(C#N)o1 Cc1oc(S(N)(=O)=O)cc1N1CC(n2cc(C3(C)CCOCC3)nn2)C1 c1(C(=O)NCC23N(C(C=CCOC)=O)CCC2CC3)ccc([N+](=O)[O-])cc1F N1(C(c2c(C)nncc2)=O)CC(F)(F)CC1CNC(c1nscc1Br)=O C1(NC(c2n(CCC)ncc2)=O)CC2CCC(C1)N2C(=O)C(C#N)C(C)C CC(C(CO)NC(C1(C)CC1(F)F)=O)NC(c1cccn1C1CC1)=O c1(C(=O)NC(CC)CN(C(=O)C(C#N)C2CC2)CC)cnc2sc(C)c(C)n12 c1(OC)cnc(Cl)cc1C(=O)NC1CC(NC(C2CC(O)C(F)C2)=O)C1 N1(CCOC)CC(C(=O)NCC(C)CNC(C2CCOC2)=O)CC1=O Fc1cc(CN2CCCC(NS(=O)(=O)C(F)(F)F)C2)ncc1Br c1(OC)cc(Br)c(CC(=O)NC(C)(Cc2cn(CCF)nn2)C(=O)O)cc1F C1(C(N(C)CCn2ccnc2)=O)CCCN1NC(=O)C1CC1 Cc1ccc(C(C)C(N2CCC(CNC(=O)Cn3cccn3)C2)=O)s1 N1(C(c2ccc(OC)nc2Cl)=O)CC2CCCC1C2CNC(C1CCSCC1)=O Cc1nc2[nH][nH]cc-2c(=NC2CC3CC(C2)N(C(=O)C=CC2CCOCC2)C3)n1 C1(C(=O)OCC)CC2CC1CN(c1cc(C(F)F)ccc1CC)C2 CC1CC(C)CN(CC(c2ccccn2)NCC2COCCN(CCC(Cl)Cl)C2)C1 C(C(C)(C)C#CC(=O)N(C)OC1CCCC1)NC(CC(C)O)=O c1(C(N(CC(C)C)CC(=O)NCC(O)CN(C)C)=O)cnn2c1CCC2 C=CCC(CC(F)F)C(=O)N(C1CN(C(=O)COc2ccc(Cl)cn2)C1)C N1(C(c2nc(C)c(C)[nH]2)=O)CC2(C1)CN(C(=O)C(C1CCCN(C)C1)(C)C)C2 c1(OCC(N2CCC(C(C)NC(=O)C(C)CN(C)C)CC2)=O)cc(Cl)ccc1Cl O=[N+]([O-])c1ccc(Cl)c(NC(Cc2ccccn2)C(=O)O)c1 C1(CNC(C2(C#N)CCCC2)=O)CN(C(c2cncnc2C2CC2)=O)CC12CC2 CN1CCC(C(=O)N(C2(CCC(=O)NOCC)CCC2)CC2CCOCC2)CC1=O CCC(C(=O)NC1(CNC(=O)CNc2ccccn2)CC(OC)C1)C(C)C C(=O)(CCCS(N)(=O)=O)NC1CCN(C(c2cc(CC(C)C)on2)=O)C1 C1(C(C(=O)NCC2N(C(C(CC)N(C)C)=O)CC(O)C2)C)CCC(C)(C)CC1 Cc1oc(Cl)nc1C(N1CC(O)(C(F)C(=O)NCC(F)C2CCC2)C1)=O n1(CCC2(C)CC2)nnnc1C(c1cnc(C2CC2)s1)NCc1ncco1 N1(C(CNC(=O)NC)=O)CCCC2CN(C(c3nc(CO)cs3)=O)CCC12 CS(=O)(=O)CCC(=O)Nc1cc(Cn2cc(-c3cc(O)no3)nn2)ccc1F C1(CNC(=O)CCC2(O)CCCC2)C(C2CC2)CCN1C(C1CC(C2CC2)C1)=O c1(CC(=O)N(CC(C)NC(=O)C(C2CCCCCC2)=O)C)ccc(O)cc1 C(=O)(C(C)=CCNC(=O)C(C1CC1)OC)NC(c1nccs1)CC N1(C(C2C(CCC)C2)=O)CC(C)C1C(=O)NC1CCN(CC(N)=O)C1 c1(C(=O)NCC2C=CC(NC(CC(CC)SC)=O)C2)cc(O)nc(O)n1 c1(C(=O)NCC(CNC(C=Cc2c(C)cncc2)=O)O)cnn2c1C(C)CCC2 C1(C(=O)NC2CCCCC2O)CCCN(C(=O)CC23CCCC2C3)CC1 c1(CCC(=O)NC2CC(NC(C3(CCCC)CCC3)=O)C2)conc1C N1(C(CC2(OC)CC2)=O)CCCCCC(NC(=O)C(O)Cc2cn(C)cn2)C1 Cc1ccc2ncc(C(=O)NCC3COCC3NC(c3cc(CO)on3)=O)n2c1 c1(C(=O)OCC)ccc(OCC(C)N(C)CC)c(Br)n1.N12CC3CC3(C1)C2=O C1(C(=O)NC23CCC(NC(C4C(C)(CC)C4)=O)(CC2)C3)CCC2(CCC2)CC1 c1(CC(C(=O)O)NC(=O)C=CC2CCCO2)cccc(F)c1 c1(CC(=O)NCCC(=O)NC2C(C(N)=O)CC2)c[nH]c2ncccc12 C#Cc1cccc(C(=O)NC2CCN(C(C3(C(F)F)CC3)=O)CC2F)c1 C(=O)(CC1COc2ccccc21)NCCOC1CN(C(CC(C)(O)C2CC2)=O)C1 C#CCC(CC)NC(c1conc1C(C)NC(=O)C(C)NC(=O)NC)=O CCC(C)CC(=O)NCC1CC(NC(C2(n3cnnn3)CC2)=O)C(O)C1 c1(C(N2CCN(C(=O)CN(CCO)CCO)C(CO)C2)=O)ncn2ccccc12 c1(OC)nccc(C)c1NC(C1(CNC(c2cc(C3CC3)no2)=O)CC1)=O N1(C(C2(C)CCCOC2)=O)C2CC1CN(C(=O)CSCC(N)=O)C2 O=C(C1=NOCC1)NCCCNC(=O)C(c1cccc(C(F)(F)F)c1)O CC1CC(C(=O)NCC=C2CCN(C(=O)C(c3ccc(F)cc3)O)CC2)=NO1 N1(C(C2CCCC(C#C)C2)=O)CCCN(C(c2cc(Cl)ccc2C)=O)C(C)C1 C1(NC(C2(CC=C)CC2)=O)CC2CN(C(c3ccc(SC(C)C)cc3)=O)CC2C1 c1(C(=O)NCCC(C)N(C(=O)CSC2CC2)C)nnc(C(C)(C)C)s1 C1(C(NOCC=C(C)C)=O)(CC)CCN(C(c2cc(C)cc(F)c2)=O)CC1 c1(CCNC(=O)Nc2n(C(C)C)nc(-c3ccccc3)c2)cc(Cl)ccc1Cl CC1CC(C(=O)NCC2(C)CC(NC(C3(CO)CCCO3)=O)C2)=NO1 C#CC1(O)CCN(C(=O)C(C)(CO)NC(=O)CC2CC(=C)C2)C1 C1(CNC(=O)OC(C)(C)C)CC(O)C(O)CC1CNC(CCC=C)=O c1(OC(C)C(=O)NC2(CNC(C3OCC3(C)C)=O)CCC2)cccc(C(C)=O)c1 n1(CC(=O)NC2C(NC(C3(c4ccc(C)o4)CC3)=O)COC2)cccnc1=O CCC(C)(COC)C(=O)NC1CCC1NC(=O)Cc1cncnc1 C(=O)(CCC(F)(F)Cn1cc(C2CCC2)nn1)N(C)Cc1c(O)ccc(F)c1Br N(C(=NCC(=O)N(C)C)NCC1CC1C)Cc1cccc(CS(=O)(=O)NC)c1 C=CCC(CC(C)C)C(=O)N1CCC2(CCN(c3cccc(F)c3[N+](=O)[O-])C2)C1 C1(c2nn[nH]n2)(NC(c2c(C)con2)=O)CCCCC1C CC1C(NC(=O)Cc2cncnc2)C(C)CCN1C(c1ccnc(F)c1)=O C1(NC(c2n(C)c(Cl)cn2)=O)CN(C(c2nc(Cl)cs2)=O)CC2(CCC2)C1 C1C(C(F)F)CC(=O)N1.c1(C(CNC(=O)OC(C)(C)C)=O)cccc(F)c1 c1(-n2c(C(CCOC)NC3CC3)nnn2)c(C)cccc1C.c12ccc(cc1)o2 CCC(CC)CC(=O)N(C)CCC1CCN(C(C23CCC(C)(C2)OC3)=O)CC1 C1(CC)CCN(N(CC2(C)CCCO2)CCCC(=O)N(C)C)CCCN1C(C)=O C(CCC(CC)CC)N(C(C(CCOC)NC(C(C)NC(CC)=O)=O)=O)C C1(CCC)CN(C(=O)Cc2cnco2)CCN1C(=O)C(n1cc(Cl)cn1)C C(=O)(C(=O)C(C)(C)C)N(C(C)C(N1CC(C)(O)C1)=O)C c1(OC)ccc(C(=O)N(C)CC2CCCC(CO)C2)nc1C C12(NC(=O)CCCCC3CC3)CCCC1N(C(=O)COc1ccsn1)CC2 c1(C(=O)NCC2CCCN(C(CCC=C(C)C)=O)C2)ccc([N+](=O)[O-])o1 N1(C(c2cnc(CNC(C(CC)(C)C)=O)nc2)=O)CCSC2(CCC2)C1 C1(C(N(C(C)C)C)=O)CN(C(c2coc(C3(O)CCOCC3)n2)=O)CCS1 c1(C(c2ccc(C)cc2Br)NC(C2CC3(CC3)C2)=O)noc2c1CNCC2 C1(NC(C(=O)N(C)C)=O)CCCCC12CCN(C(C1CC(=O)N(C)C1)=O)CC2 C1(C(C)NC(c2cnc(CC(C)(C)C)s2)=O)CN(C(C2CC=CC2)=O)CCO1 N1(C(C2(CNC(c3nc(C)oc3)=O)CCCO2)=O)CCC(C)C1C c1(OC)cc2c(cc1C(=O)NC1CC(NC(=O)C(C)C)C13CCC3)OCO2 Cc1c(N)cc(C(N2CC(NC(=O)C(C)O)CC(C)(C)C2)=O)cc1N C1(C(=O)NC2CC(NC(C3(C(F)(F)F)CC3)=O)C2)CC12CCCOC2 C1(CC)C(C(=O)N(C)Cc2cccnc2)CCN1C(C1CC(CF)C1)=O N1(C(N)=O)CCN(CCOC)CC1.CC1CC(=O)NCC(=O)NCC2OCCC12 CC(C)CC(F)(F)C(=O)N1CCC(C2CC2)(CNC(=O)C(O)CN(C)C)C1 CC1CN(C)CCC1NC(=O)C(C)(C)CCNC(C1C2CC3C(C2=O)C13)=O N1(CC)CCOC(C(=O)NC2CN(C(c3ccc(C#N)[nH]3)=O)CC2O)C1 C1(CC#C)(C(=O)NCC(CC(=O)NC)OC)CCN(C(=O)CCOCC)C1 c1(N(C)C(=O)NC2CCN(Cc3cc(C)no3)C2)nc(C(F)(F)F)c(Cl)s1 C1(C(=O)NCC2CC(F)CN2C(=O)C=Cc2cnc[nH]2)CC2CCCC(C1)C2=O C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC1(CNC(C2C(C3(C)COC3)C2)=O)CCC1 c1(C(=O)OC)cccc(N(C)C)c1C.C12CN(CC1O)Cc1ccc([nH]1)NC2=O CC(C)(C(=O)NCCOCCNC(=O)CC1CC=CCC1)C1CCCC1 c1(C(C)C)ccc(NC(C2(C)CCN(C(c3ncnn3C)=O)C2)=O)cc1Cl Cc1c[nH]cc(C(=O)N(C)CC2(O)CCN(c3nccc(CO)n3)C2)c1=O c1(C(=O)OC)ccnc2c1CN(C(C13CCCC1CS(=O)(=O)C3)=O)C2 N1(C(C=CC=CC)=O)CC2CCCC(NC(=O)C3=C(Cl)CC3)C2C1 c1(C(=O)NCC2CCCN(C(c3cc(SC)oc3)=O)C2)ccc2c(c1)CCCC2 N1(C(C(CC)CO)=O)CCOC2(C1)CN(C(C1CCC(C3CCCO3)O1)=O)C2 CN1C(=O)CN(CC(=O)N(C2CCC(NC(=O)CCC3CCC3)CC2)C)C1=O c1(CC)cncc(C(N2CCCC(C(C)(C)O)C2)=O)c1.C12(CCCO1)C(=O)NC2 N1(C(c2c(CC)non2)=O)CC(C)(CNC(=O)CC2CCCO2)CC1(C)C c1(C(=O)NCC(CC)(CC)NC(COCC(=O)OC)=O)ccn2nnnc2c1 c1(-c2nc(C)on2)cccc(C(=O)NCCNC(=O)CC2CSCCS2)c1 C12(CNC(=O)CCC3CC3)CC(CO1)N(C(=O)CCc1ccc(Cl)s1)C2 C(=O)(C(C)(CNC(C1CCCC12CCC2)=O)CC)NCCSCCOC c1(NCC2CC(C)SCC2)ncc(S(=O)(=O)NC2CC(N3CCCC3)C2)cc1Cl C1(C(N2CCC(OC)C2)=O)CC(C)(C)CCN1C(c1cscn1)=O N1(C(C(=O)C2CCCC2)=O)CCCC(N(C(C2CCC3(CC3)C2)=O)CC2CC2)C1 C1(C(=O)NC(COC)C2(C)CC2)CN(C)CCN1C(C1C2CC3C(C2)C13)=O N1(c2ncc(CC)s2)CCCCC(NC(=O)CCOc2c(C)cccc2C)C1 C=CC(CCC)CC(=O)NCC1CCCN(C(C2C3COCC23)=O)C1 CC1=NOC(C(=O)NCCn2ccc(C(=O)NCc3ccccn3)c2)C1 C1(O)(CC=C)CCN(C(=O)CCCCN(C(=O)COCC2CCC2)C)CC1 CN1CC(=O)Nc2ccc(C(=O)NCc3cc(Cl)c(F)cc3F)cc21 N1(C(C(=O)NC(C)C)=O)CC2CC(NC(C3COCCC3(F)F)=O)CC(C2)C1 C(=O)(C(C)C(F)(F)F)N(CC(C)C)CC1CCN(C(c2cc(CC)no2)=O)CC1 n1(CCC)ccc(C(=O)NC2(CCC(=O)NC(C)CCN3CCCC3)CCCC2)n1 CC1CC(=O)NC(C(N2CCCC2C(=O)NC2CCN(C)C2)=O)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1C(C)CN(C(=O)C(F)Cc2ccccc2)CC1 N1(C(C2C(C(C)(F)F)C2)=O)CC2CC(N=c3[nH]c(Cl)nc4[nH]cnc34)CC1C2 N1(C(c2ccc(OC)nc2)=O)CC2CCC1CN2C(c1c(C)nsc1C)=O c1(C(=O)NCCCC(C)NC(C=CC(CC)C)=O)cccc(Cl)c1C(F)F C(C1=NOC2CCCC12)NC(CN(C)C(C1(Cl)CCC1)=O)=O n1(CCC)nc(C)cc1C(c1nnnn1CC1CCCO1)NCC(C)(C)CC c1(C(C)(C)C(=O)OCC(=O)OC2CCC(C#N)C2)cc(F)ccc1Br N1(C(c2[nH]cc(C)c2)=O)CCN(C(C2COCCOC2)=O)C2CC12 C(N=c1[nH]c(N2CCC(CC(F)F)CC2)nc(=N)[nH]1)c1nnc(C)s1 C1(C(N(C(C)CCNC(=O)CN(C2CCCCC2)C)C)=O)CC(C)(C)OC1(C)C O(NC(=O)CC(C)C1CCCN1C(C1CCC(C)(C)CC1)=O)CCOC(C)C NC1COCCC1NC(=NCc1cnns1)NCC1CC1 N1(C(c2c(C)c[nH]c2)=O)CC(C(C)(C)C)CC(CNC(=O)C(O)Cc2cnc[nH]2)C1 N1(C(CC#N)=O)CCC(C2CN(C(c3ccc(N4CCC(O)C4)cc3)=O)C2)C1 c1(CC)nc(C#N)cc(=NCC2(NC(C3CCc4nncn4C3)=O)COC2)[nH]1 C1(CNC(C(C)=C(C)C)=O)CC2(CCC2)CN1C(c1ccccc1CC#N)=O N(C1COc2cccc(Cl)c21)C(c1cc[nH]c1C1CCC1)=O Cc1nc(O)c(Br)cc1C(=O)NC(C1CCN(C(=O)CCCF)CC1)C Cc1nc(CC(=O)NCC2CC2NC(c2noc(C3CC3)c2C)=O)c(Cl)s1 c1(OC)cc(C(=O)N(CCn2cc(-c3nccn3C)nn2)C(C)C)[nH]n1 N1(C(=O)O)CCCc2oc(Br)cc2C1.C12(CCN(CC)CC)CC(C)(CO1)C2 CCCCC(C(=O)NC1CC(F)(CNC(=O)CC2CCN(C)CC2)C1)N(C)C C1(C(N2CCC(CCN(C(CC(C)F)=O)C)CC2)=O)SC2C=CC1CC2 N1(C(C(C)NC(CC)=O)=O)CCC(C(=O)N(C)C(c2cccs2)C)CC1 c1(C(=O)NC23CC2CN(C(c2ccncc2F)=O)C3)ccc2cccnc2n1 C(=O)(CC1=CCCCC1)N1CCC(C)(C(=O)NCC(F)(F)CC2CC2)C1 N1(C(C(C2CCN(C(C3(C)CCOCC3)=O)CC2)C)=O)CCOCC(C2CC2)C1 c12cccc(c1)OC2=O.c1(C(C)=O)nccnc1C.C12CCOC1CNC(=O)N2 N1(C(C2(CF)CC2)=O)CCCC(C2CCN(C(C3CCCC(F)(F)C3)=O)CC2)C1 c1(NCCC(=O)NCC2CCCN(C(C(CSC)O)=O)C2)ccccc1[N+](=O)[O-] C1(CC=C)(NC(=O)CN(C)C)CN(C(=O)CNC(C2(COC)CCCC2)=O)C1 CC1CC=CCC1C(=O)NC1CC(CNC(c2ccc(CCN(C)C)cc2)=O)C1 Cc1nnccc1C(=O)NCC1(F)CC(NC(C2(C3CCCO3)CCCC2)=O)C1 N1(C(c2ccc(C#C)o2)=O)CCN(C(=O)CC2OCCCO2)CC1CO C1(C(N(CCC(=O)NC(CO)CCO)CCOC)=O)CCOC(C)(C)C1 C1(C)(c2nc(C)[nH]n2)CCCN1C(=O)Nc1cccc(C(C)C#N)c1 C1(C(CO)NC(C2(CC)CCOC2)=O)CCN(C(=O)CCc2cncn2C)CC1 c1(C(N(C2CCN(C(C(C)c3cccs3)=O)C2)C)=O)c(F)ccc(F)c1Cl C(c1ccccc1C)=CC(=O)NCCC(=C)CNC(c1c(C)noc1C(C)C)=O CN1CCC(C(=O)NC2C3CC2N(C(c2cnc(C4CCOC4)s2)=O)C3)CC1=O c1(C(C)NC(C(C)(C)C(C)C)c2n(CCCSC)nnn2)ccc2c(c1)OCO2 Cc1oc(C#N)cc1C(N1C2CCC1C(CNC(=O)Cc1ccns1)C2)=O Cc1cccn2nc(C(=O)NC(c3cn(CCCCCCO)nn3)(C)C)cc12 CC1(C)CC(NC(=O)CCOCC(F)(F)F)CN1C(c1ccc(F)c(CO)c1)=O C1(OC)CCC2(C(N3CCC(C)C3C(=O)NCC3=CCCC3)=O)CC12 c1(CC(=O)NCC2(O)CCCN(C(C=CC)=O)C2)c(C)nc(O)nc1C C1(c2nnnn2CCCF)(Nc2c(C(C)C)cccc2)CCCN2CCSCC12 C(=O)(N=c1cc[nH]c(C)c1C)C1CC(=C)CC1NCCN=[N+]=[N-] c1(C(N(CC(C)(C)CNC(=O)CC2CCCC2(F)F)CC)=O)c(C#N)cnn1C C1(C(=O)OC)(CNCc2cn(CC(=O)NC3(O)CCCC3)nn2)CCCO1 C(=O)(N(CCC(=O)N1CCCC1c1ccon1)OC)NC1C(CCC)C1 Cc1ccc2occ(C(=O)N(C3CCC(NC(C4OCCCO4)=O)CC3)C)c2c1 N1(C(CP(C)(C)=O)=O)CCCCCC1C(=O)NCCN1CCCCC1 C1(C(=O)OCCc2nc(-c3ccoc3)no2)CS(=O)(=O)C12CCOCC2 CCC(C)C(CC(=O)NCc1cnc(O)cc1C)NC(=O)CSC(C)(C)C N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(C2CC2)(NC(C2CCCC(=O)N2)=O)C1 c1(C(=O)NCC(CC(F)(F)F)NC(c2c(CC)nc[nH]2)=O)cc(C#N)ccc1C N1(C(c2nn(C)c(Cl)c2)=O)CCCC2CN(C(C3CC3C3CCOCC3)=O)CC12 Cc1n[nH]c(C)c1CC(=O)NC(CNC(c1cn(C2CCOC2)cn1)=O)C1CC1 N1(C(c2c[nH]c(=NC)o2)=O)CC2CN(C(C3(CC(F)F)CCC3)=O)CC2C1 C(C(CNC(=O)C(O)C(F)F)S(C)(=O)=O)NC(C1N(CC)CCCC1)=O C1(NC(C2(CCCC)CCC2)=O)CCN(C(c2cnc(CC)[nH]2)=O)CC1CC Cc1nn(C)c(C)c1C(N1CC2(CC2C(=O)Nc2cccnc2O)C1)=O CC1CCC(C(=O)N(C2CCCCC2N(C(=O)C=CC(F)(F)F)C)C)CC1 CC1(C)CC(C(=O)NC(C)(C)CNC(c2cnc(C3CCC3)s2)=O)CCO1 C(=O)(C1CCCn2nccc21)NC1CN(C(Cc2nc(C)sc2)=O)CC(O)CC1 c1(CC)ncnc(CC)c1C(N1CC2C(CNC(c3ccccc3O)=O)C2C1)=O c1(OC)ccccc1C(C)CC(=O)NCCC1CN(C(C2(F)CCC2)=O)C1 C=CCC(C)(C)CCNC(c1c(CNC(=O)CC(C)SC)cnn1C)=O C1(OC)CC(C(=O)NC2(C3CCCO3)CC2)CN(C(N(C=O)C(C)(C)C)=O)C1 CC1(C)CC1C(=O)NC1CCC1CO.C(=O)N(CCO)CCO C(CCC(=O)NC(C)C(CO)NC(=O)CCn1cc(Br)cn1)OCC=C c1(OC)cc(OC)cc(C(C)NC(C2(O)CCN(c3nnnn3C)CC2)=O)c1 CC1CN(C(c2cc(Cl)ccc2F)=O)CCN(C(C2(c3ccn(C)n3)CC2)=O)C1 C1(CNC(c2cc(OC)n[nH]2)=O)CCCN(Cc2cnn(-c3ccccc3)n2)C1 C1(CCCC)CCCC(N(C(=O)COc2ccccc2)CC)C1 C1(C(=O)NCC2C3CN(C(C4(C(=O)OC)CC4)=O)CC32)COc2ccccc2O1 C1(CC=C)(NC(c2csc(C)c2C)=O)CCN(C(=O)C(C)(C)OCCC(C)C)C1 N1(C(C(CC)OCC)=O)CCN(C(c2ccn3nncc3c2)=O)CC(C)(F)C1 CN1CC2C(C(=O)NCCn3cc(CNC(=O)C(c4ccccc4)O)nn3)C2C1 N1(C(CSCC(C)C)=O)CC(C2(NC(C3(C4CCCO4)CCC3)=O)CC2)C1 CCCC(C)CC(=O)NC1CCCC1NC(c1ccccc1CO)=O c1(CCCC(=O)NC(CNC(C(C)C)=O)C)ccc(C2CC2)cc1.C(F)(F)F C1(O)(CNC(C(N2CCC(O)CC2)C)=O)CCN(C(c2ncncc2Cl)=O)C1 N1(C(C(=C)F)=O)CCCCC(CNC(c2cc(Cl)ncc2C)=O)C1 Cc1c(C=CC(N2CCCN(C(c3ncncc3F)=O)CC2)=O)cnn1C C1(C2CCC2)(C(=O)NC(C(=O)OC)c2cscn2)CCC1 C1(C(=O)NC2(C3CN(C(C(C(=O)OC)(C)F)=O)C3)CC2)CCCC12CCOCC2 C(=O)(CC(C)(C)C(=O)OC)NCc1c(CNC(C(C(CC)C)C)=O)cccn1 C1(CNC(CCC(=O)NC)=O)CCC(C)N(C(=O)C=Cc2ccco2)C1 Cc1nccc(C(=O)NCC2(CNC(C3CCNC(=O)C3)=O)CC23CCC3)n1 C1(NC(=O)COC2CC2(F)F)CN(C(=O)C=Cc2ccncc2)C2(CCOCC2)C1 CC1CC(N2CC34N(CC(C3)C2=O)C(=O)C2C(CCC4)CC3C(C=O)C23)CCO1 Cc1cc(C)c([N+](=O)[O-])cc1C(N1CCCCC(NC(=O)C=CBr)CC1)=O C1(NC(C(C)OCC)=O)Cc2ccccc2N(C(C2CC3CCC(C2)C3)=O)C1 C(=O)(C(O)CC(N)=O)NC1C=CC(CC(=O)N(CCCC)C)C1 C1(C(=O)NC2CC(N(C(=O)CSc3cccc[n+]3[O-])C)C2)CCc2cncn2C1 C12(CNC(c3c(OC)ccs3)=O)CCC(CC1)N(C(C1(C)CCOC(C)C1)=O)C2 C1(C(N2CCC(CC#N)C2)=O)CC(C)(C)CN1C(=O)CCOC1CC1 C1(NC(C=C2CCC(C)CC2)=O)CCC12CCN(C(c1cc(C#N)cs1)=O)CC2 N1(C(c2ccc(C#N)s2)=O)CC2CCC1CN2C(c1cnc2sccc2c1)=O c1(C(=O)NC(CC)CN(C(=O)C(O)CSC)C)cc(C)sc1Br CCCC(CC)CC(=O)NC1(CF)CCN(C(c2ccc(N)c(SC)c2)=O)C1 N1(C(C2N(C(C3=CC(C)(C)C3)=O)CCCC2)=O)CCC2CCC(O)C1C2 Cc1cc(NC(C23CCCCC2C3)=O)c(C)o1 CCC(C)CCCCC(=O)NC1CCN(C(c2cnn3c2N(C)CC3)=O)CC1O CC1CN(C(C2CCOCC2)=O)CCCN1NCc1csc(N2CCCCC2)n1 c1(N2C(CC=C)CN(C(=O)C)CC2)nc(Cl)nc(C)c1Br.N1(CCC2CC2)CCCC1 c1(C(=O)NCC2(F)CCN(C(c3cc(OC)n[nH]3)=O)CC2)cnc2cc[nH]c2c1 CCC(C)CCC(=O)NC1CC(F)(CNC(=O)C(C)Cc2ccc(Cl)cc2)C1 c1(CC)onc(C)c1C(=O)NCc1nc(C(=O)NC2CCCC2CC)c(C)o1 CCC(C)C(O)C(=O)NC1CC(OCC(=O)NC(C(N)=O)C2CC2)C1 N1(C(C(c2cncnc2)C)=O)C(CC(=O)NC(CN(C)C)CO)C2CCCC12 CCC(C(=O)NCC1CCN1C(=O)Cc1csc(S)n1)n1ccnc1 N1(C(c2c(C)oc(CO)c2)=O)CCN(C(=O)CC(=O)Nc2nccs2)C2CC12 N1(C(CCOCC)=O)CCCCC2(CCN(C(c3c(C)csc3Cl)=O)C2)C1 CC1CC=C(C(=O)NCc2ccnc(C(=O)NCc3ccco3)c2)CC1 n1(CCCC(=O)NC2(CNC(C(C)=C(C)C)=O)CCOC2)c(O)nnc1O c1(NC(c2cnn(C)c2)C)ccc(S(=O)(=O)NCC2([Si](C)(C)C)CC2)cc1F N1(C(=O)NCCOCCNC(=O)CNC(C)=O)CC(CC(=O)NC)C(C2CC2)C1 c1(C(N(CCN(C(C23CC(C)C2C3)=O)CC)CC)=O)ccc(OC)c2c1CCCC2 N1(C(CC(C)C)=O)CC2COCC(C1)C2NC(c1ccc(I)c([N+](=O)[O-])c1)=O N1(C(C2ON=C(C)C2)=O)CCC(CC(=O)NCCSCC(C)C)C1(C)C C1(COC)(NC(C2CC23CCC3)=O)CCCN(C(=O)CC#N)C1 c1(C(=O)NCC(C2CC2)NC(c2csc(C(F)F)c2)=O)cncc2[nH]ccc12 C1(CNC(C2CC(OCC)C2)=O)CN(C)CCN1C(=O)CCc1cn(C)nn1 N1(C(C(C2CC2)SC)=O)CC(NC(c2cccn2C)=O)CC(C)C1 O=C(CCCCCCCO)N1CC2CC2(C(=O)Nc2ccc(O)cc2Br)C1 CCC(C)(O)C(=O)NCCCOCC(C)(C)Sc1ccccc1F C1(C(N2CCC(N(C(=O)CCCSC)CC)CC2)=O)CCC(C)C(C)C1 C1(C(N(C(CNC(C2C(=C)C2)=O)C)C)=O)(OCC)CCCCC1 c1(C(N2CC3(CN(C(c4c(OC)cc(C)s4)=O)C3)C2)=O)cc(F)cc(Br)c1F N1(C(c2ccc(C(C)=O)o2)=O)CC2CC1CN(C(=O)C=C1CCN(C)C1)C2 c1(C(=O)NCCN(CCC)C(c2cn(CCC3CC3)nc2C)=O)ncccc1C1CC1 C1(CNC(c2c[nH]nc2-c2cccs2)=O)CCCCC1NC(C1(O)CCCC1)=O N1(C(=O)N(c2nccs2)CCN(C)C)CCCC(C)(CO)C1 N1(C(C=CC)=O)CCn2ncc(CNC(C3C4CCCCCC34)=O)c2C1 N1(C(C(C=C)OC)=O)CCC(F)(C(=O)NC23CCN(CC2)CC3)CC1 CC(C)CC(O)C(=O)N(CCC(=O)NCC1CCC(C2CC2)O1)CCO C1(CNC(C2C(CNC(=O)CNc3cccnc3)C2)=O)CCSCC1 N1(C(=O)OC(C)(C)C)CCC2(CCC(Nc3ccc(C)c(Br)c3)CC2)C1 CCC(CNC(C1CCC12CCC2)=O)(CC)NC(c1csc(C(N)=O)n1)=O N1(C(C2OCCC(N(C)C)C2)=O)CC(NC(=O)CC2NC(=O)NC2=O)C(C)(C)C1 CC1CC(NC(=O)CSc2cccc[n+]2[O-])CN1C(c1cc(F)n(C)n1)=O c1(CSC2(C)N(C)CC(OC)C2)nc2c(-c3ccccn3)cccc2c(=O)n1C n1(CC(F)F)nc(CCCO)nc1-c1cc(C2CC2)on1 c1(OC)cn(CC(N2CCOC(Cc3cnc(C(=O)O)s3)C2)=O)c(C)cc1=O CCS(=O)CC(=O)NC1CCC(NC(c2ccnc(C(C)(C)O)c2)=O)C1 CN1CCC(C)(CNC(c2ccc(NC(=O)NC3CC3)cc2)=O)C1 c1(CCC)nc(C)c(NC(=O)C(=O)NC(C)(C)CC(=O)OC)s1 C(=O)(C(C)(C)C(C)(F)F)N1CC(C)CC(NC(c2c(SCC)cncc2)=O)C1 N1(C(CCCC(C)O)=O)CCC2(C1)CN(c1ncnc(C(C)(C)C)n1)C2 C=CC1(C(=O)N(C)CC=CC(=O)N(C)Cc2ocnc2C)CCOCC1 N1(C(CC2CCN(C)C(=O)O2)=O)CCC(NC(C2CCCCO2)=O)C12CC2 C(=O)(C(F)(F)F)N1C(C(=O)NCCCN2CCC2)CC1.C1CCS1 C1(N(C(=O)CC(C)n2ccnc2)CC)CCN(C(=O)CSc2n[nH]c(=N)s2)CC1 Cc1csc2ccc(C3CC3)cc12.C(=O)(C(C)(C)N(C)C)NCC1CC(=O)N1 C1(OC)CC(CNC(C2CC2F)=O)N(C(c2cnc(C3CC3)o2)=O)C1 C1(C)(CC)CC(NC(=O)C2=CCCCO2)CN1C(=O)C=C(C)CN1CCOCC1 C12(C(N3C(CNC(=O)CC4CC5(CC5)CO4)CC(O)C3)=O)CCCC1C2(F)F CCCCC(O)CCC(=O)N1CC2C(CNC(c3nc(C)sc3C)=O)C2C1 c1(NC)cncc(C(=O)NC(c2nc(NCCCn3cnnn3)co2)C)c1 N1(C(c2c(C)cc(C)o2)=O)CCC(C)N(C(=O)Cc2csc3nccn23)CC1 N1(C(C(C)NC(C)=O)=O)CCC(C(O)CNC(C23CCC2C3)=O)CC1 CC(C)C(F)C(=O)NC1CCC(N(C)C(C2CNCCO2)=O)CC1 Cc1cc(C(N2CCC(NC(=O)CNc3ccccn3)C(O)C2)=O)nc(O)c1 C=C(C)C(CC(=O)N)OCC.C1(CCC)CC(C)N(c2nc(CCC)ns2)C1 c1(C(=O)NCC2OCCN(C(Cc3nc(C)oc3)=O)C2)ccc(F)cc1C(F)F C1(C(N2CC(NC(C3(OC(C)=O)CC3)=O)C(C)C2)=O)CCC(C)=C(C)C1 c1(CC)cccc(CNC(c2cccc(F)c2)Cc2ccncc2)c1F C(=O)(CC1=CCOCC1)NC(C1CCN(C(=O)C=Cc2ccc(Cl)cc2F)C1)C c1(OC)ccc(C(=O)NCc2cn(-c3ccccc3OC)nn2)nn1 C(=O)(C(CO)C(F)(F)F)N1CC(CC(C)(C)CNC(C23CCCC2C3)=O)C1 C(=O)(C(CC(C)(C)C)OC)NC(C(=O)NCCCC=C)Cn1cncn1 N1(C(C2(C)CCC2)=O)CCCC2(CCCN2C(=O)CNC(C2CCC2)=O)C1 N1(C(c2cccc(SCCCC)c2)=O)CCCC(C)(NC(c2cnc[nH]2)=O)C1 CN1C(=O)OCC1C(=O)NC1(C)CCN(C(=O)C(c2ncc(Cl)n2C)(F)F)C1 C1(C(N(CCN(C(c2ccc(OC)c(C)c2)=O)C)C)=O)CC2C=CC1C21CC1 C(=O)(C1=CC(O)C(NC(=O)CCCC2CC2)C1)OC N1(C(c2occ(C)c2)=O)CCC(NC(c2csc(C)c2Br)=O)CC(O)C1 N1(C(C(C)NC=O)=O)CCOC2CN(C(C3CCc4nnnn4C3)=O)CC12 C1(C)(CNC(C(CCC)C)=O)COCCN(C(C2(C(F)F)CCC2)=O)C1 CC(c1ccccc1C)=CC(=O)N(CCC(C(C)C)NC(=O)CC(F)F)C C1(CNC(C(CCSC)O)=O)CC(F)(F)CN1C(c1ccc(F)cc1C)=O N1(C(C(C)OC2CCCCC2)=O)CCC(N=c2[nH]cnc3cnccc23)C1 O=C1CC2C(C(=O)OCCC(F)F)C2C1 C(=O)(C(C)C(=O)NC1CC(C)(C)C1)NC(C)(C)C.N1(C(COC)=O)CCC1C(=O)OC C(=O)(CC(C)C(C)C)N1CC(N(C(C(CC)NC(c2ccco2)=O)=O)C)C1 c1(CNC(c2c(C)cc(F)s2)=O)n[nH]c2c1CN(C(C1CC1F)=O)CC2 c1(C(N2CC(CCCNC(C3(C)CCC3)=O)OCC2)=O)nc(O)nc(O)c1F N1(C(C(C2CCN(C(C)=O)C2)C)=O)CCN2CCC1C2 Cc1nc(O)ccc1C(=O)NCc1ocnc1C(N1CCC(n2ccnc2)C1)=O CN1CCCC(N=c2ccnc(N3CCC(Oc4ccncc4)C3)[nH]2)C1 CCC(C)C(C)(O)CNC(=O)CCC1(C)CN(C(=O)C(C)(C)C#N)C1 Cc1cc(C(N2CC3C(NC(c4cc(F)cnc4Cl)=O)C3C2)=O)cc(F)c1 C12(CNC(CCOCC#C)=O)CCC(CC1)N2C(c1cnco1)=O C1(C2CN(C(c3ccnn3CC3CCOC3)=O)C2)(NC(C2CCC(=O)O2)=O)CC1 N(C(=NCCC1CC1)N1CCC(OC)CC1)CC1C(OC(C)(C)C)CC1 c1(C(=O)NCC2C(CNC(C(CC#C)O)=O)C2)nn(C)c(C)c1Cl C(C(C)(C(=O)N1CCCCO1)NC(C1CC(F)C(=O)N1)=O)OC C=C=CCCC(=O)N1CCC(C2CCCCN2C(C2CCCC2)=O)CC1 C(=O)(CCCC(=O)N(C)C)N1CC2C(NC(Cc3n(CC(C)C)ncc3)=O)C2C1 N1(C(CN2CCC(C)C2)=O)CC(CNC(=O)C=Cc2nccs2)C2(CC2)C1 N1(C(C(C)OC(C)(C)C)=O)C2CCC1CC(NC(c1ccnc(C(N)=O)c1)=O)C2 C(=O)(CC(C)(C)C(=O)N1CCC(CNC(=O)CCc2nncs2)(OC)C1)OC c1(N(C(C)=O)C)ccccc1C(=O)NCCC(O)CNC(C1CC(CF)C1)=O CC#CCCC(=O)NCCN(CCCCCC)C(C1CC(F)(F)CS1)=O Cc1nc2c([nH]1)CN(C(C1CCN(C(=O)C(O)CC(C)(C)C)CCO1)=O)CC2 C1(NC(c2ccc(OC)cn2)=O)CC(NC(c2ccc(F)cc2F)=O)C12CCC2 c1(C(C)C)cccc(C(=O)NC2CC2CNC(=O)C(C)N(C)C)c1N C(=O)(C1=C(C)CCCC1)N(CCN(C(c1cncc(OCC)c1)=O)CC)CC c1(C(=O)NCC(CCCC)NC(C2CC(CN(C)C)C2)=O)cc(F)ccc1C C(=O)(CCCCC(C)CC)NCCOCCNC(CC(C=C)(C)C)=O c1(C(=O)NCC2N(C(C(CC)=O)=O)CCOC2)n[nH]c2c1CCC2C CC1CN(C(=O)C=Cc2ccc(Cl)cc2)CCC1NC(c1coc(N(C)C)n1)=O c1(C(=O)NC2C(NC(c3cc(C)nn3CC(F)(F)F)=O)C2)ccc(C)cc1O C1(CNC(C(C)(O)C2CCC2)=O)CCN(C(C2CCCC23CC3)=O)CC1O N1(C(=O)Cc2ccc(F)cc2)CC2CC1CC2NC(C1CC(F)(CO)C1)=O C1(C(F)(F)F)(NC(=O)CC2CC2)CC(C(F)F)(N)C1.C(C=CCNC(C)=O)=CC C(=O)(C(C)CC(=O)N1CCCC(C(=O)OC)C1)OC.C12(CNC3CC3)CCN(CC1)C2 c1(CNC(C(N2CC(C#C)N(C)CC2)=O)=O)ccc2c(c1)OCCO2 N1(C(CC#C)=O)CC2CN(C(c3cc(C(=O)OCC)ccc3C)=O)CC12 C12(NC(CNC(C(CCOC)OC)=O)=O)CCC(CC1)C2(C)C.C(CO)O C1(C)(NC(C2(NC(C3COCC(C)O3)=O)CC(O)C2)=O)CCCC1(F)F CC1(CNC(c2ccc(Cl)nc2Cl)=O)CCCN(C(c2ccnn2C2CC2)=O)C1 C1(C(=O)NC(C)CC(C)N(C(C=CCC)=O)CC)CCCN(C(C)CC)C1 N1(C(C2CCC(C)(C)OC2)=O)CC2CC1CN(C(c1cc(C(F)F)[nH]n1)=O)C2 CN1CCc2c(sc(NC(C3C(O)CC3O)=O)c2C#N)C1 C1(CC(=O)NC2CCCC(NC(CCCNC(=O)OC)=O)C2)CCCC(C)(C)C1 C(=O)(C(C)CC(C)(C)C)NCCOC1CCN(C(Cc2c(C)cc(C)s2)=O)C1 N1(CC)CCOC(C(N2C(C(N3CC(c4ncc[nH]4)C3)=O)CC3CC23)=O)C1 C1(C(=O)NC2(CNC(CCC=CC)=O)CC2)CCCC(C)CC1 c1(C(N2CCCC2c2ccncn2)C(=O)NCCSC)cnc(Cl)s1 C(=O)(C(C)CC(C)(C)C)N1C(C(=O)NCC(C(C)C)C)CC1 CC(C)(C(=O)NCCCOC1CCN(C(c2cnc(S)nc2)=O)CC1)C(F)(F)F Cc1cc(C(N2CCC(F)CC2)C(=O)NCC2CCCO2)n2nccc2n1 C(=O)(C1Cc2ccc(F)cc21)N(C1CC(NC(c2nccnc2O)=O)C1)C c1(C(N2CCCC(NC(C(CO)N(C)C)=O)C2)=O)nn(C)c(C(F)(F)F)c1Cl Cc1ccsc1C=CC(N1CC2(NC(=O)C(N3C(=O)CCC3=O)C)CC1C2)=O C=CCCCCN=c1[nH]c(N2CCC(F)(F)C(COC)C2)nc2ccc(OC)cc12 c1(C(=O)NCc2cc(C)sc2C)nc2cc3c(cc2s1)OC(F)(F)O3 C1(CC)C(NC(C2CCC(F)(F)C2)=O)CCN1C(=O)CN(C(C)C)C1CC1 c1(C(=O)NCCN(C(C2CCCC2C(F)F)=O)CC)ccc(S(N)(=O)=O)o1 CCCCCCCC(=O)N1CCN(C2(C3CC3)CCNC2)CC1 C1(C(=O)NC(C=C)(C)C)COCC1NC(=O)C=C(C)C(C)(C)C Cc1cc(C(=O)NCC2CCCC(CNC(=O)CCN3CCCCC3)C2)[nH]c1C C12(NC(C(C3CCN(C(COC(CC)C)=O)C3)F)=O)CCC(CC1)C2 c1(OC)ccc2[nH]c(=NC3CC(=C4CC4)C3)nc(N3CCOC(C4CC4)C3)c2c1 N1(C(C2(CC)CCN(C(c3cc(O)n(C)n3)=O)C2)=O)CCCC2(CCC2)C1C N1(CCNC(CCNC(COC)=O)=O)CCN(C(=O)CC2CC(C)OC2C)CC1 N1(C(C2CC(SC)C2)=O)CC2CCC(C1)N2C(C1CCC(O)C1)=O N1(c2n[nH]c(=NCc3c(F)cccn3)o2)CCCC(C2CCC2)CC1 c1(C(C(=O)Nc2nnc(CCOC)s2)(F)F)nnc2n1CCCC2 C1(C(N2CC(CNC(c3n(C=C)ncc3)=O)C2)=O)CC2COCC(C1)C2 C1(CCNC(C(C2CCCC2)OC)=O)CC(C)=NO1.C1(=O)CCOCCN1 Cc1nc(C)c(-c2nc(-c3cc(C)oc3C)nn2C2CCCCC2C)[nH]1 C1(CNC(COC(C)=O)=O)CC12CCN(C(c1csc(-c3ccoc3)n1)=O)CC2 c1(C(N2C(CCNC(C(C)SCCCC)=O)CCC2)=O)cccc(CO)c1 C1(CCNC(=O)C(F)=C2CCCC2)CCCCN1C(=O)CN1C(=O)CNC1=O c1(CCC(=O)NC(C)CCCNC(C2(N(C)C)CC2)=O)nc2ccccc2[nH]1 C1(CNC(C(C)(C)F)=O)CN(C(C2CC2C2CCC2)=O)CCC12CCC2 C(=O)(CCCC#CC)N(CC1(O)CCN(C(CCOCC#C)=O)C1)CC CCCCCCCC(=O)NC1CN(C(=O)COc2cnn(C)c2)CC1C C1(NC(c2ccc(C3CCC3)nc2)=O)CCCC12CN(C(c1csc(Cl)n1)=O)C2 c1(OC)ccc(Cl)c(C(=O)NC2CCC(NC(c3ncccc3OC)=O)C2)n1 N1(CCNC(=O)C2=CCC2)CCC(NC(c2ccc(OCF)cc2)=O)CC1 N1(C(C(c2cc3ccccc3o2)C)=O)CCCC(C)(C)C1C#N N1(C(C2(C#N)CCCC2)=O)CC2CCCC(C1)N2C(C1CC1C(F)(F)F)=O C1(C(N(C(CC#C)C)C)=O)CN(C(c2cccnc2O)=O)CCC1(C)C N1(C(C(COC)OC)=O)CC2CC(NC(=O)C=C)CC2C1.c1(O)ccc(F)c(Cl)c1 c1(C(N(CC(C)CNC(C2CC(CF)C2)=O)C)=O)cccc(CC2CCCO2)c1 C12CCCCN1C(=O)C(=O)NCCC(C(C)C)NC2.c1(CC)cn(C)[nH]c1=N c1(OC)cc(C(F)(F)F)[nH]c(=NC(C)CNC(=O)C(C)C2CCOC2)n1 N1(C(C2CN(CC)C(=O)N2)=O)CC2(CCN(C(c3ccccn3)=O)CC2)C1 CCC(C)C(=O)C(=O)N1CCN(C(c2cc(C3CC3)on2)=O)CC1 c1(C(=O)NC(CNC(c2cc(C#N)no2)=O)CO)cccc(C#CC2CC2)c1 C1(NC(CN(C2CC3(C2)CC(N)CCO3)CC)=O)C(C)(C)CCCC1(C)C c1(OC)cc(CC(=O)OC(c2cn(CCO)nn2)C)cc(F)c1F N1(C(C2N(CC)CCC2)=O)CCN(C(=O)CCCN2CCCC2)CC(C)(C)C1 C#CC1(C(=O)NCC(CC=C)OC)CN(C(=O)Cn2nc(C)oc2=O)C1 Cc1cn2c(C(=O)N(CC(O)CN(C(=O)CC(C)N(C)C)C)C)cnc2s1 C(C)(CO)(C(=O)N(C)CCC1CCN(C(=O)C=CC2CCCC2)CC1)OC CC#CCCCC(=O)N1CC2CC1CN2C(=O)C(C)NS(=O)(=O)c1cccs1 C(CCCCCC)(c1n(CC=C)nnn1)NCc1cnn(CC)c1 C1(CC(N)=O)CCCN(C(=O)NC(c2cccc(Br)c2)C2CC2)C1 C1(CCNC(c2cnc(C)[nH]2)=O)CCN(C(C2CCC(=O)N2)=O)CCC1(F)F c1(C(=O)NC(C#C)CC)conc1CNC(=O)CC1CC2CC2C1 CC(O)C(C)C(=O)NC1CCCC1NC(C1(c2ncccc2F)CC1)=O C1(CNC(=O)CSC(C)C)CC(O)C1.CCC(C)N(C(=O)CC1CC1)C c1(N2CC(C)=C(C)CC2)nc(C)cc(=NCc2csc(-c3ccn(C)n3)n2)[nH]1 c1(C(=O)NC(CN(C(c2ccc(NC)cn2)=O)C)C)c[nH]c2c(C)c(C)ccc12 CC(C(=O)N(C1CC1)CC1CCCN1C(c1cc(C2CCC2)on1)=O)S(N)(=O)=O c1(CCC(=O)N(C)CCNC(c2ccc(-c3cc[nH]n3)s2)=O)cc(F)ccc1F CC1CN(C(C2(C)CCCS2)=O)CC1CC(=O)NCC(c1cn(C)cn1)O CN1N=C(CC(=O)NCC2CCN2C(c2cc3c(cn2)CCCC3)=O)CC1=O C1(NC(c2ccn(C(C)C)n2)=O)COCCC1NC(C1CCN1S(C)(=O)=O)=O C1(c2cn(C3CC(NC(CCCS(C)(=O)=O)=O)C3)nn2)(N(C)C)CC(F)(F)C1 N1(C(C(CC)C(=O)OC)=O)CCN(C(=O)C(C)(C)CSC)C2(CCC2)C1 c1(C(=O)NCC2CC(NC(c3c(C)cc(O)nc3)=O)C2)cnc2n1C(C)CCC2 c1(C(=O)NC2(CCNC(CN(C)C3CC3)=O)CC2)cnn2c1OCC(F)C2 C1(NC(C2CCCN(CC)C2)=O)CN(C(=O)CC#N)CC2(CCOCC2)C1 c1(C(=O)OC(CCN(C)CC)=O)cc2nc(C3CC3)cc(COC)n2n1 Cc1cncc([N+](=O)[O-])c1N1CCC(CNC(c2cc(Cl)n(C)n2)=O)C1 CC1OCCCC1C(=O)NC1(CNC(C2CCCN2N=O)=O)CCC1 N1(C(c2c(NC(C)=O)cccn2)=O)CCCN(c2ncc(F)c(SC)n2)CC1C c1(C(=O)NCC(C)(C2CC2)NC(C(CC(C)(C)C)O)=O)cc(F)c(F)c(C#N)c1 N1(C(CN2CCC(C)C2)=O)CCCC(N(CCF)C(c2cc[nH]c2)=O)C1 CC(CCCCNC(=O)CNc1cccnc1)NC(c1nc(=O)n(C)[nH]1)=O Cc1ncnc(C)c1C(=O)NC(C)CN(CC(=O)NC1CCC(C(N)=O)CC1)C N1(C(C(=O)OC(C)(C)C)(C)C2CN(C(=O)OCC)C2)CCC2NCCCC2C1 C(C)(C(C(C)C)NC(C1CC(n2cnnc2)C1)=O)NC(c1nc(CC)oc1)=O c1(CCC)ncoc1C(=O)N(C1CCCCC1)CCNC(=O)CN1CC=CC1 C(=O)(C1CCCc2scnc21)NC1C(NC(c2c(C(C)C)ocn2)=O)COCC1 c1(C(=O)NCCOCCNC(CC(C=C)CC)=O)c(C)c2ccc(F)cc2oc1=O C1(OCC=C)CCN(C(=O)CCCNC(C23CSCC2C3)=O)C1 C1(CCC)CN(C(c2cnc(OC)nc2)=O)CC1NC(=O)C(C)(C)CF C1(C(=O)NCCN(C(=O)Cc2csc(S)n2)C2CC2)CC(c2ccccc2)=NO1 C(c1ccc(OC)c(C)c1)=CC(=O)NC1CC(CNC(C=CCOC)=O)C1(C)C C1(C(=O)NC(CCC)C)CC12CCN(C(C1C(C)(C)C1(C)C)=O)CC2 CC(C(=O)N(CCCNC(=O)C(C)C1CCC1)C(C)C)=C1CCCC1 Cc1cc(C)c(C(=O)NC(CO)C(C)NC(c2ccc(=O)oc2)=O)c(S)n1 c1(C(=O)NCC2CC(NC(C3C(C)CCC3)=O)C2)cc(Br)cc(F)c1O c1(C(C)NC2CC(C(C)NC(=O)COC(C)(C)C)C2)ccc(F)cc1 C(=O)(C1CCSc2ccccc21)NCC(C)N(C(c1cc(OC)c(C)cc1)=O)C Cc1c(Cl)ccc(C(=O)NCC2CN(C(C3(C(C)C)CC3)=O)CC2C)c1N N1(C(C(CCC)=CCC)=O)CCCC(NC(c2ccc(OC)c(O)c2)=O)C1CC c1(CCCN=C(NCC(=C)CC)NCCF)c[nH]c2c(Br)cccc12 C1(C(N2CC3(CN(C(c4nc(C)oc4)=O)C3)C2)=O)CC2COCCN2C1 N1(C(C=CCOC)=O)CCN(C)CC1CNC(=O)CC(C)(C)SC CCCN(OC)C(=O)C(c1cccs1)N(C(c1ccc(Cl)o1)=O)CC c1(C(N2CCC(O)(CCNC(c3c(CC)cns3)=O)C2)=O)ccc2nncn2c1 CC(C(=O)N1CCC(O)(CCNC(c2ccc(C(F)(F)F)cc2)=O)C1)C(C)(F)F c1(C(N)=O)cnc(Cl)[nH]c1=NC(CNC(=O)C1Cc2ccc(F)cc21)C1CC1 CC1CN(C(c2ccco2)=O)CCC1CNC(c1cc(Br)cnc1N)=O CC1CCN(C(=O)CC2COCCO2)CC1CNC(C1CCC(F)CC1)=O C1(CNC(C(C)C2(O)CCC2)=O)CCC(NC(=O)C=C2CCSCC2)CC1 C1(C(=O)NC2CCC(CC(=O)N(CC(C)(O)C3CC3)C)C2)(CC)CCOC1 C1(OC)CC(F)CN(C(C2CN(C(=O)C(F)(F)c3ccccc3)CCN2)=O)C1 C1(CN(C(c2cn(CCC)nc2C)=O)C)CN(C(=O)C(C)(C)CCF)CC12CC2 N1(C(C2CCC(N(C)C)C2)=O)C2CCC1(CNC(=O)CC1=CCCC1)CC2 c1(OC)nn(C)c2nc(C)cc(NC3C4C5CC6C3C6C45)c12 CCC(CC(=O)NCC1COCCN(C(=O)C=C2CCN(C)CC2)C1)C(C)(C)C c1(C(=O)NC2C(NC(C(C)(C)OC(C)=O)=O)CC2)cnc2[nH]c(C)nc2c1 N1(C(C(=O)NC2(C)CC2n2cnc(-c3ccccc3)c2Br)=O)CC2(CCCCC2)C1 c1(CC)cnc(Cl)[nH]c1=NC1CC(NC(C2CCC(C)(C)O2)=O)C1 C=CC(C)(O)C(=O)NCCC1CCN(C(=O)C(CC)OC)CC1 N1(C(c2cc(C)c(Br)o2)=O)CC(NC(C2CCCC2C2CC2)=O)C(C)(C)C1 C(=O)(C(O)CCC(C)(C)N)NCC(=O)NC(CC(C)C)CO c1(SC)cnn2ccccc12.C12(c3ccccc3)CN(C1)C(=O)NCc1nc2on1 c1(OC)cccc(C(N2CCCC2CCNC(c2cc(C)c(C)[nH]2)=O)=O)c1 N1(C(CC(C)(C)SC)=O)CC(F)(F)CC1(C)CNC(=O)Cn1cccn1 C1(C(=O)NC2CC(CC(=O)NCc3ccc(Cl)o3)C2)CCNC1=O N1(C(c2c(CC)sc(=N)[nH]2)=O)CC(O)C(O)C1CNC(c1coc(COC)n1)=O C(CCCCC(=O)N(C)C(c1ccco1)C)NC(c1cc(C(C)C)no1)=O c1(OCCOC)cnc(NC(=O)NC(Cc2ccc(OC)cc2)C)nc1C(C)C CC1CCC(C)N1CC(=O)NCc1cccc(C2CN(C(=O)COCCF)C2)c1 c1(C(N2CC(O)(CCNC(CCC=C(C)C)=O)C2)=O)c(C)cccc1N C#CCC(CC(F)F)NC(C1(F)CCN(C(=O)C2=CCCCC2)C1)=O c1(C2N(C(CS(C)(=O)=O)CO)CCC2)nc2ccc(Cl)cc2o1 c1(C(=O)NC(CC2CN(C(CCC(=O)OC)=O)C2)C)c(F)cc(Cl)cc1F c1(C(C(N2CC(NC(=O)CC(F)F)C(O)C2)=O)O)ccc(Cl)c(Cl)c1 C(=O)(C1=C(Cl)CCCC1)N1CC2C(CNC(CCc3c(OC)cccc3)=O)(C2)C1 Cc1sc(C(=O)NC(CNC(=O)C(C)OC2CCCCC2)C(C)C)c(C)c1C c1(C(=O)OC)ccc(Cl)c(SC)n1 C1(C)(NC(C2C(C)=C2)=O)CN(C(=O)CC(O)C2CC2)C1 C#Cc1ccc(C(=O)NC2CN(C(C3(O)CCC(C)CC3)=O)CCC2C)cc1 N1(C(c2occ(C)c2)=O)CCC(N(C(=O)CC2CC(C)OC2C)C)CC1 Cn1cc(-c2nc(-c3ccccc3)nn2Cc2cccs2)c2ccccc2c1=O c1(SC)ccc(C(N2CC(NC(c3csc(Br)c3)=O)C2)=O)o1 CC1(C)COC(C(N2CCC(NC(=O)CNC(c3ccccc3)=O)CC2)=O)C1 C1(O)(CC)CCCN(C(=O)C(CNC(=O)C(C)NC=O)OC)C1 c1(NC(=O)N(C)CC2(SCC)CC2)cc(I)nn1C Cn1cnc2c(NC(c3ccc(-c4ccc(O)c(CO)c4)cn3)=O)ncnc12 C1(C)(CNC(CC(C)F)=O)CN(C(c2ccc(-c3cn[nH]c3)cn2)=O)C(C)(C)C1 c1(OC)ccc(C(N2CCC(NC(=O)C(C(C)(C)C)N(C)C)C(O)C2)=O)c(F)c1 c1(OC)cc(C(N2CCC(N(C(=O)C(O)C(C)SC)C)C2)=O)c(Cl)cn1 C(=O)(N=C1C=CC=C1C(F)(F)F)C1OCCN(Cc2scc(C)c2)C1 C1(NC(C2CN(C(COCCCOC)=O)CC2C)=O)CCN(C)CC1C#N CN=c1nc(N2CCCCC(C)C2)[nH]c(=NC(C)CCC(F)(F)F)[nH]1 n1(CCC(=O)NCCCN(C(C2CC2C(F)F)=O)CC)ccccc1=O C=CC1OCCC1C(N1CCCC1CC(=O)NC(C)C(=O)OCC)=O Cc1cn2c(n1)CCC(CNCC13CCCCC(NS(=O)(=O)Nc4ccccc4)(C1)C3)C2 C1(C(C)C)CN(C(c2cn(CC(F)(F)F)cn2)=O)CCC1NC(c1cccs1)=O CCC(C)(C)C(O)C(=O)NC1CCN(C(c2ccc(C(F)(F)F)o2)=O)CC1(C)C C1(NC(C2CC(NC(CC)=O)C2)=O)CN(C(C2C=CCS2)=O)CC1C(F)F C1(Cc2cn(C(COCC)C(=O)NCC(C)(C)C(F)(F)F)nn2)CCc2ncnn2C1 N1(C(C(c2ccc(C)s2)C)=O)CCN(C(c2cccc(O)c2C)=O)C(C)C1 C1(C(=O)NC(CNC(c2c(C(C)C)nn(C)c2)=O)C)CC2(C1)CC1(CC1)C2 C1(C(N(C(C)CN(C(=O)Cn2cnnn2)C)C)=O)CNC(=O)N1 N1(C(c2ccccn2)C)CC2CCCCC2(C(N2CCC(c3ccco3)C2)=O)C1 Cn1c(C(=O)NCC2(NC(=O)CNC(=O)NC3CC3)CC2)cc2sccc12 c1(C(N(CC(C)NC(C2(C(C)(C)OC)CC2)=O)C)=O)cccn1C C(=O)(C1=Cc2cc(CC)ccc2OC1)NC(CNC(CCC(=O)OCC)=O)CC C12CN(C(=O)OC(C)(C)C)CC1C(=O)N2.C1(=O)CN1.N(C)(CCO)CC N1(C(CSCC)=O)CCC(C(=O)Nc2cncc(OC)c2)C1(C)C c1(C(=O)NC2C(CNC(C(c3cncn3C)OC)=O)C2)ccc(CC#N)cc1 Cc1cnc2n1CCC(C(=O)Nc1cccc(-c3cn4ccsc4n3)c1)C2 c1(OC)ccc([N+](=O)[O-])c(NCC(C)NC(=O)C(C)(C)NC(C)=O)c1F C(=O)(C(C)(C)C(F)(F)F)N1CC2(CC(CNC(CC3CCC(C)O3)=O)C2)C1 C(=O)(C1=NN(c2ccccc2)C(=O)CC1)NC(C)CNC(C1CC(C)(CO)C1)=O Cc1ccsc1C(=O)NCC(C(=O)N(C)CC1(F)CCCC1)N(C)C N1(C(C=CCN(CC)CC)=O)CC(OC)CC(NC(=O)C(CCC)OC)C1 c1(C(N2C(C(C)C)CN(C(C3(O)CC3)=O)CC2)=O)cc2ccc(Cl)cn2c1 N1(C(C2(C)CCC2)=O)CCOC2(CCCN(C(c3cccnc3Br)=O)C2)C1 CCC(CCOC)C(=O)NCC(CNC(c1sccc1OC(F)F)=O)OC C1(NC(COCCCC)=O)CCN(C(C2CCCC2C2CC2)=O)CC1CC c1(OC)cc(OC)c(N)c(C(=O)N(C)CC2CCN(C(=O)CSC)C2)c1 N(C1c2ccccc2CC1NC(c1ccccc1O)=O)C(CCC#C)=O N1(C(CCC(C(=O)OC)NC(=O)OC(C)(C)C)=O)CCCC2(CCSCC2)C1 C(=O)(CCCCC(C)(C)C)NC(CSCC)C(N1CCS(=O)CC1C)=O C=CC(C)C(C)C(=O)NCc1ccccc1-n1cc(C(=O)OC(C)(C)C)nn1 c1(NC(C2N(C(c3ccc(OC)o3)=O)CC2)=O)cnc(N2CCCCC2)nc1 Cc1nc(Br)n(C2CCN(c3ccc(OCC(F)(F)F)cn3)C2=O)c1C c1(CCC(=O)N)cccnc1.C12CCCN1CC=CCC2(C)O.c1(N)cc(Cl)no1 c1(C2(C(=O)NCC3CCC(NC(C(C)(O)C4CC4)=O)C3)CC2)cccc(Cl)n1 c1(C(=O)NCC(CNC(C(c2cccs2)SC)=O)CO)cc(C#N)ccc1F c1(OCC)nc(N2CC3C(CNC(C4CCN(C)C(=O)C4)=O)C3C2)ncc1C N1(Cc2cc(C(=O)OC)ncc2)CC2C(NC(C3(C(F)(F)F)CC3)=O)C2C1 c1(CNC(=O)C(N2CCCC(CC3CC4(CCC4)C3)C2)=O)ccccc1F N1(C(c2c(C)n[nH]c2C)=O)CC2CCC(N(C(=O)CSc3cnn(C)c3)C)C2C1 C1(CC=C)(C(=O)N(CC(C)SC)C)CN(C(=O)CC(C)C2CC2)C1 CCCC(C)(C)CC(=O)NC1(CNC(c2ccnc(Cl)c2O)=O)CC1 c1(C(=O)NCCC2CCCN(C(C=CC(CC)C)=O)CC2)cccn2nncc12 CCC(CC)C(C)C(=O)NC(CNC(=O)C=Cc1cc(F)cc(F)c1)C(C)C C1(NC(c2cccc(C)c2)=O)CCN(C(c2ccc(C)[nH]2)=O)CC1C N1(C(COC(CC)C)=O)CC(NC(c2cnn(C)c2C)=O)C(n2cccn2)C1 c1(C(=O)NCCC(C)N(C)C(C2C3COCC23)=O)cnc2c(c1)CNC2=O N1(C(C=CC(CC)C)=O)CC(O)(C2(CNC(=O)C(CC)Oc3ccccc3)CC2)C1 N1(C(C(=O)Nc2scc(-c3ccc(C)c(C)c3)n2)=O)CCOCC12CCOCC2 CC1CN(C(c2ccnc(O)c2)=O)CC1NC(=O)C(C)(C)C1CCCCO1 c1(C(N2CCC(N(C)C(c3ccnc(S)c3)=O)C2)=O)cccc2cnnc(O)c12 c1(CC)cc(O)nc(N2CCCC(C(=O)N(CCOC)Cc3cccs3)CC2)n1 Cc1cccc(C)c1C(=O)N(CC(C)NC(=O)C(F)(F)c1nccs1)CCSC N#Cc1cncc(C(N2CCNC(C(N3CCC4(CC3)CC4)=O)C2)=O)c1 C(CNC(=O)CC(C)(C)C1CC1)(C(C)C(C)C)NC(C(c1cc(C)sc1)(C)C)=O CCC(CC)CCCNC(=O)CC1CC(C2CC2)C1 c1(C(=O)NCC2C(C(=O)NC(c3ncc[nH]3)C)C2)csc(CO)n1 CC(CC(=O)NC12COC(C1)C(NC(=O)CCN1CCCCCC1)C2)C(F)(F)F N(C1CCc2c(Br)cccc21)C(N1Cc2c(C)csc2C1)=O C1(CNC(=O)CC2CC(c3ccccc3)C2)CN(C(c2cnco2)=O)CCCO1 CCCCC(C(=O)NC1(C)CCN(C(c2ccsc2-n2cnnn2)=O)C1)C(C)C CCC(CNC(=O)C(C)(C)C(C)NC(C1CC1CCOC)=O)(CC)CO C(CN=c1[nH]c2c(c(=NC(C)C3CCOCC3)[nH]1)CCCC2)NC(CC)=O C(C(C)(C)C(=O)NC1CN(C(=O)C=CC(C)C)CC1n1cccn1)NC(C)=O c1(C(N2CC(O)CC(NC(C=CC)=O)C2)=O)cc2cccc(F)c2o1 C1(COC)CN(C(=O)CSCC(=O)OC)CCN1C(C1CN(S(=O)(=O)CC)C1)=O C1(NC(=O)CCCF)CC2(C1)CN(C(c1cc(C3CC3)cs1)=O)C2 Cc1ccc(F)c(CNC(C2CSCCN2Cc2ccc(Br)cc2I)=O)c1 CC1CC(C(=O)N(C(CNC(C2(Br)CC2)=O)C2CC2)C)C1 c1(C(C)C)nnc(C=CC(=O)NC(C)(C)C(C)NC(=O)C#CC2CC2)o1 C#CCCCCCC(=O)N1CC2(C1)CN(C(c1cc(C)n(CC)c1C)=O)C2 c1(OCC)ccc(F)c(C(N2CCC(NC(C3CC3COC)=O)C(F)C2)=O)c1N CCC(C)C(=O)C(=O)N1CC2(CC2)CC1CC(N1CCC(C(C)O)CC1)=O C(=O)(C1CCCc2cncn21)N1CC(CC(C)NC(c2c(C(C)C)nns2)=O)C1 O=C1CC2(C1)CC(C(N1CCC(F)(C(N3CCCCC(CO)C3)=O)CC1)=O)C2 CN1CC2OCCN(C(C3(NC(=O)C(O)C(F)(F)F)CC(O)C3)=O)C2C1 N1(C(CNC(CCC)=O)=O)CC(C)(NC(C2(C(=O)Nc3cn(C)nn3)CC2)=O)C1 N1(C(=O)CCC2CCC2)CC(C2CCCN(C(C3(C4CC4)CC3)=O)C2)C1 N1(C(C(CCC)N(C)C)=O)CCCC2(CCN(c3nc4ccccc4s3)CC2)C1 c1(NC(=O)Nc2n(CC)nc(C(C)(C)C)c2)nc2c(O)ncnc2s1 c1(OC)ccc(F)cc1C(=O)NC1(CF)CN(C(c2occc2C2CC2)=O)C1 c12cccnc1NCCOC1CCN2C1.c1(CC(=CC(=O)OC)C)ccccc1 C#CCC(C)(C(=O)NC(CO)C(O)CCC)NC(=O)Cc1ccc(O)cn1 C1(CC(=O)N(CC(C(C)C)C)C2CC2)CCC(C)N(C(=O)C(c2cnn(C)c2)=O)C1 N1(C(c2cc(OCC)n[nH]2)=O)CC(O)CCC1C(=O)N1CCCCO1 N1(C(c2n(C(C)C)ncc2Cl)=O)CC2CN(C(c3cnc(C(N)=O)s3)=O)CC2C1 CC1CN(C(c2nccn2C)=O)CCC1N(C)C(C1(NC(N)=O)CC1)=O CC(CN(C)C(C)C)N=c1[nH]c2c(ncn2Cc2ccccc2)s1 S(=O)(=O)(C1COCC1F)NC(C1C(C(=O)OC)C1(C)C)=O Cc1noc(C)c1C(C)C(N1CCCC(N(C(=O)Cn2cnnc2)CCO)C1)=O c1(C(=O)NCC(C)N(C(C(c2cccc(Cl)c2)CC)=O)C)c(C)ccc(C)c1N CCCCC(O)CC(=O)N1CC(F)(F)CC1CNC(=O)Cc1cccnc1Br N1(C(C2(CNC(Cc3c(C)nccc3)=O)CC(C)(C)C2)=O)CCN(C)C(C)C1 c1(C(=O)NCC2CCN2CCCc2c(F)cccc2Cl)coc2c1C(O)CCC2 C=CC(CCC)CC(=O)N1CCN(C)C(C(N2CC(N(C)CC)C2)=O)C1 c1(N2CC(CO)CC(C)C2)ncccc1S(=O)(=O)NCC(c1cn(C)cn1)O CC(C)(C)C(C(=O)NC1CC(CCNC(C2CC3(CC3)CO2)=O)C1)NS(C)(=O)=O Cc1ccc([N+](=O)[O-])c(NCC(O)CNC(C2CCc3nnnn3C2)=O)c1 N1(CC2C(C)CCCC2)C(=O)CCN(CCCc2nnnn2C)C1=O c1(C(N2CC(O)(C(=O)NCC(=O)NC(C3CCCCO3)CC)C2)=O)cnc(C)n1C CCC(C)(C(=O)NCC1CC(C)N(C(=O)C2=COCC2)C1)C(N)=O c1(NC(=O)CCCN(C(C23CC(c4ccccc4)C2C3)=O)C2CC2)cncc(Br)c1 C1(NC(c2nnn(C)n2)=O)CC(F)CN(C(=O)CC2(C)CCS(=O)(=O)N2)C1 C1(NC(CCCCCC=C)=O)COC2(CCCN(C(=O)CC3CCCC3)C2)C1 c1(C(=O)NC2C(C(=O)Nc3cc(C(N)=O)ncc3)CCC2)cnn2c1NCCC2 CC1CCc2nc(C(=O)NC3CC(C)(NC(c4ccc(F)c(Cl)c4)=O)C3)cn2C1 C(=O)(C1=Cc2ccccc2OC1)NC(Cc1cccc(OC)c1)C C1(CNC(C=C(C)Cl)=O)CC2CC2N1C(=O)CC1CSCCO1 C(=O)(CCCCCc1ccccc1)NC(CNC(CN(C1CCCC1)C)=O)C(C)(C)C C1(NC(C(C)(C)SC)=O)CN(C(=O)CN(C)C(c2ccccc2)=O)CC12CC2 CC1(C)C2CCC1(C(=O)NC1(CCNC(C3CC4CCCC4C3)=O)CCC1)C2 C1(CCNC(=O)C=Cc2cnc[nH]2)COCCN1C(c1cnn(C2CC2)c1)=O c1(C(N(CCN(C(=O)Cc2cncn2C2CC2)CC)CC)=O)ccnn1CCF c1(CNC(=O)NC(c2c(Cl)cccc2Cl)CO)cc(Br)ccc1F Cc1cc2c(C(N3CC(=O)NC4(CCC4)C3)=O)nccn2n1 C12(NC(C3CCC(CC)O3)=O)CCC(CN(C(C3CN4CCC3CC4)=O)C1)C2 S(=O)(=O)(c1ccc(Cl)cc1)NCC(=O)NC1C(CNC(CC(C(C)C)C)=O)CCC1 CN1CCN(C(=O)CCCC#N)CC1C(N1CCC(CO)C1(C)C)=O C1(C(=O)NC2(C)CCN(C(=O)CC3CC4(CC4)CO3)C2)CC2(CCOCC2)C1 c1(-c2ccc(-c3nc(COC)n(C4CS(=O)(=O)C4)n3)nc2)ccnc2ccccc12 c1(C(=O)NC23CC2CNC3)ncnc2c1ncn2-c1ccccc1F.C12(CC1)CC2 c12ncccc1C(=O)NC2.C1(C(N2CCC2CO)=O)(SC)CCC1 C1(NC(C=Cc2cn(C)nc2)=O)CCN(C(C2C3CCCC23)=O)CC(O)C1 c1(C(N(CCC(C)NC(c2cc(CC)nn2C)=O)C)=O)cc(N)cnc1Cl CC1CC2(CC(C(=O)N(C3CCN(C(C4CC(n5cccn5)C4)=O)C3)C)C2)C1 n1(C(C)C(=O)N(CC(O)CNC(=O)COCC(F)F)C)ccc(C2CC2)n1 n1(CC)nc(C)c([N+](=O)[O-])c1N1CCN(C(c2cccc3c2OCO3)=O)CC1 c1(C(N2CC(O)(CNC(=O)Cn3ncccc3=O)C2)=O)c[nH]cc(Cl)c1=O N1(C(C=C(CCN(C)C)Cl)=O)CC(NC(=O)CC2CCCC23CC3)C(O)C1 C1(N(C(c2nnc(S)n2C)=O)SCC)CCCN(C(=O)COCCC(C)C)C1 c1(CNC(CCN(C(=O)CCC2CCCO2)CC#C)=O)cn(CC)nn1 CON(C)C1CCN(C(C23CCC(CC2NC(c2ccccc2F)=O)C3)=O)CC1 C1(CNC(CCC(=O)OC)=O)C2CCC(C2)N1C(C12CC(CC(C)O1)C2)=O N1(CCCCCNC(=O)CCc2ncccn2)CCN(C(=O)Cc2cocn2)CC1 N1(C(C(CC)(F)F)=O)CCOC2(CCN(CCOCC(F)F)CC2)C1 N1(C(COC(C)C)=O)CC(NC(C2CCOC2c2nccn2C)=O)CC12CCC2 CC(C)CC(C)CC(=O)N1CC(C2(Nc3ncccc3C#N)CC2)C1 c1(NCCC(C)(C)F)nc(=NCc2n[nH]cc2Br)[nH]c2c1COC2 C(=O)(C1=CCOCC1)NCC(CCOC)NC(=O)C(C)c1cccs1 N12CCCC1C2C.c1(OC(C)C)ccnc(CO)n1 C=CCCC(CC(C)C)C(=O)NC1(C2CCCN(C(C3CNC(=O)N3)=O)C2)CC1 Cc1nnc2c(C(N3CCOC(C(C)NC(=O)COCC(F)F)C3)=O)cccn12 c1(NC(N(CCC)Cc2ccc(C)cc2)=O)ccc2nc(C(F)(F)Br)[nH]c2c1 c1(C(=O)NC(C(C)NC(CCCCOC)=O)(C)C)ncn2c1CCCC2 CC1(C)CC(CNC(=O)CCC(=O)c2ccncc2)CN1C(C1CC1C(N)=O)=O C1(C(=O)NCC(C)CNC(=O)CCSCc2ccccc2)CCC(O)CC1 N1(C(c2ccc(S(N)(=O)=O)s2)=O)CCC(NC(=O)CC(O)C2CC2)C2(CCC2)C1 c1(C(C(F)F)NC(C)CSC(C)(C)C)ccccc1 C(c1ccc(C(F)F)o1)=CC(=O)N(CC(C)NC(=O)COCC1CCCO1)C C1(C(=O)NCC23CC2CN(C(=O)CCCn2cccn2)C3)CC2C=CCC(C1)C2 CN1CCCCC1CC(=O)NC1CCN(C(c2cncn2-c2ccccc2)=O)C1 C1(C(=O)NCC2N(C(CC3(COC)CC3)=O)CCCC2)CCc2n[nH]c(C)c2C1 C(C(C)(C)C#CC(=O)NCc1cnc(C(C)C)[nH]1)NC(C1C=C(C)CS1)=O C=CC(F)(F)C(=O)N1CCCC(N(C(c2csc(C(N)=O)n2)=O)CC)C1 C1(C(=O)OC)CCCC(F)C1.c1(CCCC)ccc(C2c3n(nnn3)C3(CC3)N2)s1 c1(OCC)cc(F)ccc1C(c1nnnn1C1(C)CC1)NCc1ccccc1C Cc1c(C(=O)NCC23CCC(CC2)CO3)n(C)c2ccccc12 C(=O)(C1=NNC(=O)C1)NC1CC2C(NC(c3c(CC)occ3C(F)(F)F)=O)C2C1 c1(SCC)cc(C)ccc1-c1c[nH]nc1C(=O)NC(C)C.c12c[nH]c(c1)NC2=O Cc1nc2ccc(Br)cn2c1C(=O)N(C)CC1CCN(C(=O)C=CC(C)C)C1 C1(C(N2CCN(C(=O)C=C3CCC3)CC2)=O)(OC)CCCN(Cc2ccccc2)C1 C(=O)(C1=CCCCO1)NCc1cc(C(=O)NCc2c(CC)noc2C)n(C)n1 C(=O)(CCC1=CCCCC1)NC(C(=O)N(CC(=C)C)C)CC(=C)Cl N1(C(COCC#C)=O)CC(CNC(c2cnc(C)nc2C)=O)OC(C)(C)C1 C1(NC(CCc2cn(C)nc2)=O)CC(NC(C2CC2C#N)=O)CC1O CCC(CC(=O)NCC1(C(=O)NC2CCOC(C)(C)C2)CC2(CC2)C1)C(F)F N1(C(c2cccc(C#C)c2F)=O)CCCC2CN(C(=O)CN(C)C)CC12 C(N=c1cc[nH]cc1[N+](=O)[O-])C1CCN(C(c2cc(C)sc2C)=O)CC1C S(=O)(=O)(c1ccsc1C#N)NCC(C)(CO)OC Cc1c[nH]c2ncc(C(=O)NCCNC(=O)C3=NOC4COCC34)cc12 N1(C(C(=CC2CCCC2)C)=O)CCC(C)N(C(=O)CSCc2cscn2)CC1 CC1CCN(C(C2CC(=O)CCO2)=O)CC1CC(=O)NC1CCCC1F N1(CC(=O)NC2(CNC(c3ncc(C)nc3)=O)CCOCC2)CCCCCC1=O C(CC(C(C)(C)C)NC(C1CCCO1)=O)N(C(Cn1c(C)csc1=O)=O)C N1(C(=O)Cc2ccsc2)CCN(C(c2cnc(O)c(Cl)c2)=O)C(C2CC2)C1 CC#CCC(C(=O)NCC1CC1(F)F)NC(=O)Cc1ccc(O)cn1 C=CCC(C)N=c1nc2ncn(C)c2c(N2CCC(Nc3ccnc(C)n3)C2)[nH]1 N1(C(c2c(C)scn2)=O)CCOC(C(N2CCCC2C(C)C)=O)C1 C1(CNC(C=CC(CC)=CC)=O)CCC(C)N(C(c2ccco2)=O)C1 C=CC(CC)CC(=O)NCC(CNC(=O)C(F)(F)c1nccn1C)OC N1(C(CC2(C)CC2F)=O)CCC2(CC1)CCN(C(=O)COC1CCOC1)CC2 CCC(C)(C)C(O)C(=O)Nc1ccc(-c2ncccc2OC(C)=O)c(F)c1 CC(F)(C(=O)NC1CC(NC(C2CC2c2cncs2)=O)C1)c1ccccc1 C1(C(=O)OC)CCCC1F.C1(=O)NCCN1 C1(NC(C2(CCC)CC2)=O)CC(OC)CN(C(=O)C(CC)OCCOC)C1 C(=O)(C1=CCCN(C(C23CCC(CC2)C3)=O)C1)N1CC(N(C)C)C2(C1)CC2 C1(CC)CN(C(C2(C#N)CCC2)=O)CCC1NC(c1cncnc1CC)=O c1(C(=O)NCC2C(NC(CCOC)=O)CCC2)cnncc1OC C(C(C(C)C(C)C)NC(c1sccc1CN(C)C)=O)NC(CCC)=O c1(CCOC)nc(=NC(=O)N2CCC(C3CCCO3)CC2)s[nH]1 C(=O)(C(CC(C)C)ONC(c1cnccc1C#N)=O)N(CC)CC1CC1 CC(CN=c1nc(N2CCOC(COC(C)C)C2)c2[nH]ccc2[nH]1)c1ccsc1 CC1CCCC2C(=O)N(C3CCc4nc(N(C)C)ncc4C3)C(=O)N2C1 C=CCC(CC)C(=O)NC1(CNC(=O)CCCSC)CCOC1 N1(C(CCC)=O)CCCC(C(C2CC2)NC(=O)C=C2CCC(C)C2)C1 c1(C(N2CC(CC(=O)NCC(C)N(C(COC)=O)C)C2)=O)ccc(C)o1 CC1CN(C(=O)C=CCF)CCN1c1cc(-c2ccccc2)ncn1 Cn1ccnc1CC(=O)NCCCOCCNC(C1(F)CCOC1)=O c1(OC)cc(F)c(F)cc1NC(C1CC(F)CN(CC2CC2F)C1)=O CC1C(NC(c2cnc[nH]2)=O)CCCN1C(c1cccc(N(C)C)n1)=O C1(NC(CCSCC)=O)CC(C)CN(C(c2cc(C3CC3)ccc2Cl)=O)C1 c12ccnc(n1)SC1CC(C1)NC2C.c1(C(=O)OCCO)ccnn1C N1(C(=O)CS)CCCN(C(N2CCCC2)=O)CC1.C1(C=O)CC1(F)Cl C12(C(N3CC(COC)N(C(c4cnsc4)=O)CC3)=O)CC3CC(C1)CC(C)(C3)C2 c1(CCC(=O)NC(CNC(C(C)(F)F)=O)C2CC2)ccccc1C#N C(=O)(CCCC(CCC)CCC)NCCCCCN(C(C(C=C)(C)C)=O)C C1(C(=O)NCC2(CNC(C3(CC)CC3(F)F)=O)CC2)OCC2CCCC1C2 c12cc(n(C)n1)CNC2=O.C1(CNC(CCOCCC)=O)(OC)CCOC1 C(=O)(C1=CC(C)(C)C1)NCC=C(C(=O)NC(C#C)CC(C)C)C c1(C(N2CC(CCNC(c3cnc(O)s3)=O)(OC)C2)=O)ncccc1C(C)(C)C C#Cc1cccc(C(=O)NC2CN(C(c3cnc(C)cn3)=O)CCC2(C)C)c1F C(=O)(C#CC1(C)CCCO1)N1C2CN(C(c3ccn(C)n3)=O)C(CC2)C1 N1(C(C(CC2CC2)OC)=O)CCC(C(=O)NC2CCCC2)(OC)C1 N1(C(CC(=O)OCC)=O)CCC2CCCC12C(=O)NC(C)Cc1cccnc1 Cc1cc(C)c(C(=O)NC2CC(CCNC(C3CCN(C)C3=O)=O)C2)c(O)n1 N1(C(c2nc(CCCC)sc2)=O)CCN(C(=O)C(C)OC)CC1c1cn[nH]c1 c1(NC(N(CC)Cc2ccc(F)s2)=O)c(Br)ccc(Cl)c1F C1(C(N2CCC(C(C)C)(CO)C2)=O)CCC(C)N(c2nccnc2C(C)(C)C)C1 C(=O)(C1CC(=O)c2ccccc21)N(CC(C)NC(c1cc(C)c(C)nn1)=O)C N1(C(C(C)OCC2CC2)=O)CC(C)CN(C(C23CC(C)(CO2)C3)=O)CC1C c1(C(=O)NC2CC(NC(C(CC(C)C)N(C)C)=O)C2)cc(F)c(Br)cc1F c1(C(=O)NCC2CCCS2(=O)=O)cccc(S(=O)(=O)C(F)F)c1 N1(C(CCNC(N)=O)=O)CCC(NC(=O)CCCNC(N)=O)CC1 c1(OCC(=O)NCCCN(C(=O)Cc2ncncc2Cl)CC)cccc(C)c1 CC(C)C(F)(F)CC(=O)NC1CCC1NC(=O)C(O)CC1CCCC1 C1CCN(CC(=O)NC2CC=CC2)CC1.C12CC(C)N(C1)C(=O)N2.NC(=O)C1CC1 C=C=CCCC(=O)NCCOCC(C(=O)NC(C)(CO)CC=C)N(C)C C(CCO)(C(F)(F)F)NC(C(C)N(CCC)C(C1CCCSC1C)=O)=O N1(C(c2c(OC)n[nH]c2)=O)CCC(CNC(c2ccc(C(N)=O)nc2)=O)C(O)C1 N12CC(C3(CC3)C1)CC1(CC(=C)C1)C2=O.C1(C(=O)OC)CN(C2CCC2)C1 C1(O)(CCNC(c2c(C)nc(O)s2)=O)CCN(C(c2ccc(=O)n(C)c2)=O)CC1 N1(C(c2c(C)n(C)cc2)=O)CCC2CN(C(c3c(F)cc(F)cc3Cl)=O)CC2C1 c1(C(N(CCNC(CC2(C#N)CC2)=O)C2CC2)=O)ccc([N+](=O)[O-])cc1Cl C=C=CC(C)C(=O)NCC(c1ccc(C(C)C)cc1)NC(c1ccc(C)cc1)=O C1(NC(C2(CSC)CC2)=O)C2CC3C(C2)C13C(N1CCCC(F)(F)C1)=O C(C1=CCN(C(c2ccnnc2O)=O)CC1)NC(C1N(S(C)(=O)=O)CCC1)=O C1(CNC(CSCc2cccc(C)c2)=O)CN(C(=O)CCCC2CC2)CCC1O C1(NC(CC(C=C)C)=O)CCCCCCC1NC(=O)C(CC)N(C)C N1(C(C2(OC)CCN(C(C3CCS3(=O)=O)=O)C2)=O)CCC2C(O)CC12 c1(C(=O)NCC(C)(C)NC(=O)CNS(C)(=O)=O)cccc(C(C)(C)C(F)(F)F)c1 c1(C(N(CCCCCC(=O)NCC2CCCC2(C)C)C)=O)c[nH]c2ncccc12 CC(C)CC(C)(CO)NC(C1CC2(CC(NC(=O)CC3CC(N(C)C)C3)C2)C1)=O C(CCC(C(=O)NC1CCN2CCC1C2)NC(=O)C=CC1CCC1)OC Cn1cc(C=CCNC(C2C(NC(=O)COc3ccsn3)C2)=O)nn1 CCCCCCC(F)C(=O)NC(C)CCNC(c1cc(F)c(N)cc1F)=O Cc1oc(C(=O)NCc2cc(C(=O)NC3CCOC3C)n(C)n2)cc1CO N1(C(c2c(C)nc(CC)o2)=O)CC2CC1CN(C(C1CC3(CCCCC3)C1)=O)C2 C1(NC(c2ccc(OCC)cc2)=O)CCN(C(=O)CCC#N)C(C2CC2)C1 N1(C(C(C)Cc2cccc(F)c2)=O)CC2CC(CNC(=O)CCC3(C)CC3)C2C1 C12(NC(c3cc(Cl)c(Cl)nc3Cl)=O)CCCC1N(Cc1ccc(Cl)nc1)CC2 CC1(C)C2CN(Cc3cc(-c4ccc(-c5ccc(F)cc5)cc4)cnc3F)CC12 N1(C(C2(OC)CCCC2)=O)CC2CC2(CNC(c2ccncc2F)=O)C1 C1(N(C(c2c(C)nsc2)=O)C)CCN(C(=O)CCc2ccccc2O)CC1C C12(CO)CCC(C(=O)N(CC(CC)NC(=O)CCC(=O)OC)C)(CO1)C2.CCO C1(C(=O)NCC2N(C(c3ccc(C)c(C)c3)=O)CC2)CCCC2(CCC2)O1 c1(C(=O)NCC2(NC(C3CCCN3C)=O)CC(OC)C2)ccc(F)cc1F c1(OC)ccc(C(=O)NC2C(C(N3CCC4(CC3)CC4)=O)CC2)c(N)c1 C1(NC(C2CCCN(CCC)C2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1C C(=O)(C(O)CC(C)C)N(CCCC(=O)OC)CC.c12nnc(o1)C2.c1(SC)ccccc1 C(=O)(C(CC(C)(C)C)NC(c1ncnc(C)c1C)=O)N1CCCC(OC(C)C)C1 c1(OC)csc(C(=O)OCC2CCN(C3CCN(C)CC3)C2)c1OC c1(NCCCCN(C)C(C2CCCCN2C(=O)CC2CC2)=O)c(F)ccc(=O)o1 c1(CN2C3C(C(=O)OC)CC(C3)C2)cc(=O)n2[nH]cnc2n1 c1(CC)cccc(C(C(=O)NC(c2cccc(Cl)c2)C)NCC(CSC)CO)c1 O=S1(=O)CCN1.c1(CC(c2cncs2)NCC(F)F)ncccn1 N1(C(CCCCSC)=O)CC(NC(c2ccc(C)c(CO)c2)=O)CC12CCCC2 CCCCC(C)(C)NC(=O)CCC1CCCCN1C(C1CC(=O)C1)=O C1(NC(C2(C)CC(C)(C)C2)=O)CCC(C)(C)CC1CNC(c1cc(Cl)ccn1)=O C(=O)(CCS(N)(=O)=O)NC1(CC=C)CCN(C(C2CCS(=O)(=O)N2)=O)C1 N1(C(C(CCC)C)=O)CCC(C(=O)NC(C(N)=O)C2CC2)CC1(C)C C1(NC(C(CC=C)CC)=O)CC2CCC(C1)N2C(C1OCCCO1)=O c1(OC)c(CC(N2CCCC(C)C2CCNC(=O)C=CSC)=O)cccc1F C1(NC(COCC(=O)NC)=O)(COC)CCN(C(=O)CN2CCC(C)CC2)C1 Cc1cc(=NCc2cncs2)[nH]c(N2CC(=O)NC(C)(C(C)C)C2)n1 C(C(CC(C)C)C(=O)N1CC2CCC1(CNC(=O)Cc1cccs1)CC2)OC C(c1cnc(C(C)(C)C)s1)=CC(=O)NCC1C=CCN1C(C1CCCCO1)=O c1(CC(=O)NC2CCCN(C(Cn3c(C)ccn3)=O)C2)c[nH]c2ncccc12 Cc1cccnc1CC(=O)NCC(C1CCC1)NC(=O)CC1(OC(=N)O)CC1 CC1CN(C(c2c(C3CC3)cnn2C)=O)CCC1CNC(=O)Cn1ncnn1 CCC(C)(C)C(O)C(=O)NCC(C1CCC1)NC(c1cccn1C1CCCC1)=O C(=O)(C1CCCc2c[nH]nc21)NCC1(CNC(=O)Cc2cnns2)CC1(F)F C1(CNC(c2ccc(C)nc2O)=O)CN(C(C2CS(=O)(=O)C2)=O)CC(C)(C)C1 N1(C(C(CC=CCC)C)=O)CC(C(=O)NC2CCOCC2OC)CCC1(C)C CC1COC(C)(C)CN1C(=O)C(CCC1CC1)NC(=O)CC#N n1(CC(N2C(CNC(C(=O)NC(C)C)=O)CC(C)(C)C2)=O)cc(S(C)(=O)=O)cn1 C=CCC(C(=O)NC1CCCCC1N(C(=O)C=CC(C)(C)C)C)OC CC1=C(C(=O)N2CCN(C(=O)CC3COC(C)(C)CO3)CC2C)CCCC1 c1(NCCN(CC(c2cc(C)no2)OC)CC)ccc(F)cc1 c1(C(=O)NCCOCCN(C(C2CN(C(=O)NC)C2)=O)C)cc2cnccc2o1 C1(NC(C(=O)NCc2c(C)cc(C3CC3)o2)=O)CCC2(CCCC2)C1 n1(CC)cc(CN2CCC(CC(=O)NCCC3(CCC(=O)O)CC3)C2)c(C)n1 N1(C(CC(C=C)C)=O)CC(C2CCCN(C(=O)Cn3ccnn3)C2)C1 c1(C(N(C2CCN(C(=O)C=CCO)C2)C(C)C)=O)ccsc1C#N C1(C)(CCNC(c2n(C)cnc2)=O)CCN(C(c2ccc(C(F)(F)F)s2)=O)C1 N1(CCN(CC)Cc2ccccc2)CCOCC1C.c1(N)sc(S)nc1C N1(C(=O)C=C(Cl)Cl)CCCC2(C1)CN(C(=O)C(O)Cn1cncn1)C2 N1(C(CC(CN(C)C)C(F)F)=O)CC2(CCCN(C(C3(C)COC3)=O)C2)C1 Cc1cc(C(=O)NCC2CC2NC(c2c(C(F)F)n[nH]c2C)=O)c(Br)s1 CC1=C(C(=O)NCC2CCCC2NC(c2cc(F)ncc2C)=O)CCC1 N1(C(C(c2cccnc2)NC(=O)CC(=O)NC2CC2)=O)CC2(CCOC2=O)C1 C1(CNC(C(CCOCC)C)=O)CN(C(c2ccc(Cl)cc2Cl)=O)CC(C)(C)C1 C12(NC(C3CCCSC3)=O)CCC(CN(C(C3CCCC4(CC4)C3)=O)C1)C2 CC1CC(NC(C2(N(C)C)CCCC2)=O)CCN1C(=O)C(O)C1CC1 c1(C(=O)NC(CN(C(c2ccoc2)=O)CC)C)cc(C2CC2)on1.S(C)(=O)(=O)N C=CCCCCCCC(=O)NCc1c[nH]nc1C(=O)NC(CO)C(=O)N(C)C Cc1ccn(C)c1C(N1CCCC(NC(C2CCN2C2CCCC2)=O)C1)=O Cc1cc(C(N2CCC(N(C(=O)CC3COCC3O)CCO)C2)=O)cs1 C(=O)(C(C)(C)C(C)O)N1CCC(N(CC(=O)NC(C)C)C)C1 c1(NC)cc(Cl)ccc1C(=O)NC1(C)CN(C(=O)COCc2ccccc2)C1 c1(OC)nc(N(CC(=O)NC2CC3CCC2C3)C)nc2[nH]cnc12 C1(C(C)C)CC1C1CN(C(c2ccc(OC(C)C#N)cc2)C(=O)NC2COC2)C1 c1(CCC(=O)NC(CC)CNC(=O)Cc2cc[nH]c2)cccc(Cl)c1 Cc1occc(=O)c1OCC(N1CCCC1C(C)NC(=O)CCC(C)(F)F)=O c1(C(N2CCC(CNC(=O)Cc3ccncc3Cl)C2)=O)cnc2c(c1)CCC2 C(=O)(C(O)C(CCC)NC(=O)C=CCCC)NCCCCC#CC Nc1cccc(-c2cn(CCCNC(C3CC3c3nc(C(=O)O)cs3)=O)nn2)c1 C(=O)(C(O)CSC)NCCSCC(=O)NCCCOCCC(=O)NC c1(Nc2cccc(C(=O)OC)c2)cccc2c1CC(NC(=O)OC(C)(C)C)C2 N1(C(c2cncc(C(C)(C)C)c2)=O)CCC(NC(C2CCCNC2=O)=O)C(O)C1 CC1CN(C(c2ncnc(O)c2F)=O)CC(C)N(C(c2c(F)cccc2F)=O)C1 c1(C(N2CCC(N(C(CNC(c3c(C)onc3)=O)=O)C)C2)=O)cn(C)nc1C C1(NCc2cccc(C(=O)OC)c2)CCN(c2ncnc(CO)c2OC)CC1C C1(C(=O)NC(C)(C)CNC(c2cc(Cl)ccc2C(F)F)=O)CCc2cncn2C1 c1(CN2CCCC(NC(Cc3cccc(OC)c3)=O)C2)c(Cl)cc(OC)cc1Cl C1(C(N)=O)C=CCN(C(C2CCCN2C(=O)CN2CCSCC2)=O)C1 C1(N=c2ccc(-n3cccn3)n[nH]2)(C(=O)OC)CC(OC)C1 N1(C(CCC2CCCN(C(CSCC(=O)OC)=O)C2)=O)CCC2(CCO2)C1 CC1OCCC1(C)C(=O)NCC(C)(C)NC(c1cn(C2CCCCC2)nn1)=O N1(C(CCOC)=O)C(CNC(=O)C(Cc2ccccc2)SC)CC2CCCC12 C(=O)(C1(C)CCn2ccnc21)N1C(C2CCN(C(C(C)OC)=O)CC2)C(C)(C)C1 C1(CC=C)(NC(C2CC2CC)=O)CN(C(=O)C(C)NC(=O)NC)C1 C1(C(=O)NCC=CCNC(c2ccc(CSC)o2)=O)CC2(C)C1C=CN2C C1(C(C)C)CCN(C(=O)C=CCC(C)(C)NC(C2(C)CC3CC3C2)=O)CC1 N1(C(CC2(OCC)CCOCC2)=O)CCN(C(=O)C(C)CN(C)C)C2COCC12 c1(C(N2C(CNC(C(CCC)NC(N)=O)=O)CC2)=O)c(F)ccc(F)c1Cl C1(CC(=O)NCC(CNC(=O)COCCCN=[N+]=[N-])OC)CCC(C)CC1 N1(C(C2(OCC)CCCC2)=O)CCC(NC(c2cnn(C)c2Cl)=O)CC1C C1(CC)CN(C(C2CCC(=O)N2)=O)CC1NC(c1ccnc(OC)c1)=O C1(NC(C(c2n(C)cnc2)O)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)cn1)C2 N1(C(c2nc(C(C)OC)oc2)=O)CCCCC1CNC(C1CCOCC1)=O C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CC(OC)CN1C(c1cc(O)cs1)=O c1(C(N2C(C(C)(C)NC(C(C)CO)=O)CCC2)=O)n[nH]c2cc(Br)ccc12 N1(C(C(F)=CCC)=O)CC2CCCC2(NC(=O)Cc2cccc(C)c2)C1 c1(C(=O)OC)ccc2c(c1)N(CCN=c1ncc(F)c[nH]1)CCO2 C1(C(=O)NCC(C(=O)OC)(C)O)CNC(=O)CN1C(=O)C=Cc1cncs1 C1(C)(C(=O)NCCC(C(=O)OCC)C)CC(F)(F)CN1C(=O)OC(C)(C)C C1(N(C(=O)C(F)CC2CCC2)C)CS(=O)(=O)C1(C)C.C1(=O)CC(=O)N1 c1(C(N2CC(CNC(C(C)(C)C(N)=O)=O)C(F)(F)C2)=O)nccc2cccnc12 N1(C(CC2(OC)CCCCC2)=O)CCCC(F)(CNC(C2(Cl)CC2(F)F)=O)C1 C1(NC(CC2N(C(CC3CCCC(=O)N3)=O)CCCC2)=O)C2CCCC1CC2 N1(C(N)=O)CCCC(C(=O)NCC2C3CC2N(C(=O)CC2CCS(=O)(=O)C2)C3)C1 c1(OC)ccncc1C(N1CCCC1CC(=O)N(C(CC1CC1)CO)C)=O c1(CC(=O)NC2(C(=O)NCCC3CC(SC)C3)CCC2)ccc(F)c(Br)c1 C(=O)(CCN=c1[nH]ccs1)N1CC(C)(CNC(=O)CC2C=CCCC2)OCC1 CCC(CC)CC(F)C(=O)NC(C1CCCCC1)CNC(=O)C(C)N=[N+]=[N-] C1(c2cn(C)nc2)CC(CNS(=O)(=O)CCCC2CC2)CCO1 C1(NC(C(C)O)=O)CC2CCC(C1)N2S(=O)(=O)C1CCOCC1 C(=O)(C(C)CC(C)C(C)=O)NCCC1(C(=O)NC2C(C#C)CCC2)CC1 N1(C(CNC(C(N2C(COC)C(C)(C)C2)=O)=O)C)CCc2ccccc21 c1(C(=O)NC2C(CNC(c3csc(O)n3)=O)CCC2)c(F)cccc1F c1(C(=O)NC(C(C)NC(c2cc(Br)nn2C)=O)C)cnc2cnn(C)c2c1 N1(C(c2cc(COC)no2)=O)CCC2(CCN(C(c3cccnc3)=O)C2)C1 N1(CC(=O)OC)CCN(C(=O)C(N2CCSC(c3ccccc3)C2)C)CC1 C1(C(=O)OCC2(CCC=C)CC2)CN(C(=O)NC(C)(C)C)C1.NC Cc1ccc(CCC(=O)NCCCNC(=O)Cc2cccc(Cl)c2)cc1F C1(OC)CC(CNC(c2ccc(CNC(C3CC(C)(O)C3)=O)o2)=O)C1(C)C N1(C(C2CC(OC)C2)=O)CC(CNC(c2ccc(O)c(F)c2F)=O)CC12CCC2 C1(CC#C)(C(=O)NCC(C)OCCO)CCN(C(C2CN(C)C2)=O)C1 n1(CC)cc(C2CN(C(=O)Nc3sccc3COC(=O)CC3CC(F)C3)C2)nn1 C(C(O)C(F)(F)F)NC(C(C)(C)CCNC(=O)CCOC1CCCC1)=O.OC CCCS(=O)(=O)CC(=O)NC1CN(C(=O)C(C)C(C)n2cccn2)CC1(C)C C1(CNC(C(c2ccccc2)C)=O)CN(C(c2nccc(Cl)c2O)=O)CCN1C N1(C(c2c(CC)cco2)=O)CCC(C(C)NC(c2ccoc2Cl)=O)CC1 CCCCCCNC(=O)CC1(CNC(=O)C(C)COCC)CC1 C1(OC)CC(C(=O)NCc2cn[nH]c2)N(C(C2CC3C=CC2C3)=O)C1 c1(-c2cn(CC(=O)OC)nn2)cccc(C)n1.C1(F)(C(N2CC2)=O)CCOC1.CC O=C1CCN(CCOc2ccc(Cl)c(Cl)c2)C(=O)N1CC1CCC2CC12 C1(C(=O)OC)CC2OCCC2N1C(C1COC(C)(C)C1)=O C(C)(C)(CC(=O)NC(CC1CC1)C1CC1)N(C(CC1ON=C(C)C1)=O)C c1(C(=O)NCC2C(NC(=O)CC3CCCC3)CC2)ccc2c(c1)COC2 C1(CC=C)(NC(c2nnn(C)n2)=O)CCN(C(C2CCCCC2C(C)(C)C)=O)C1 c1(C(=O)NCC2C=CC(NC(C(C)(C)F)=O)C2)ccccc1Cn1cccn1 N1(C(c2c(C#N)scc2)=O)C(C(=O)NCCOC(F)(F)C(F)(F)F)CCC12CC2 Cc1cccc(CC(=O)N(C(C)CNC(c2cnc(O)n2C)=O)C)c1 c1(C(N(C)CC2CCN(C(CCCN(C)C)=O)C2)=O)ccc([N+](=O)[O-])cc1F N1(C(CC2C(CC)CC2)=O)CC2CC(C)N(C(c3ccc(OC)cc3)=O)C2C1 C1(C)(CNC(CC2(OC)CN(C(C3CCCCC3O)=O)C2)=O)CC2(CCC2)C1 N1(C(c2c(C)n(CC(F)F)nc2)=O)C2CCC1CC(NC(c1c[nH][nH]c1=N)=O)C2 c1(OC)cnc(C(=O)NC2CC2NC(C2CCN(C(=O)N(C)C)CC2)=O)c(F)c1 c1(NC(C)C(N2CC(CC3CC3)C(C)C2)=O)cccc(Cl)c1 N1(C(=O)NC2C(Cl)(C(=O)OC)C2)CCOC(C)(C(=O)OC(C)(C)C)C1 C1(NC(=O)CCc2cnc[nH]2)C2CCC(C2)C1C(=O)NCC(c1ccccc1)O c1(OC)cncc(NC(C2CC2C(C)NC(c2csnc2Cl)=O)=O)c1.C1C(=O)N1 C(=O)(C(C)(CO)NC(C1CC(C)CC1)=O)N(CCOCC#C)C C(=O)(CC(C)OC)NCC(CC)NC(=O)Cn1nccc1C N1(C(CC2N(C)CC=CC2)=O)CC2(CCCC2NC(=O)CCC(N)=O)C1 c1(OC)ccc2[nH]c(=NCC(F)F)nc(N(C)CCc3sc(C)nc3C)c2c1 c1(C(CNC(c2cc(Cl)no2)=O)NC(C(F)OC)=O)ccc(F)cc1F c1(CC(N2CCCC(C)(CNC(=O)CCCF)C2)=O)csc2c(F)cccc12 CCC(C)C(C(=O)NCC#CC(F)(F)F)N(C)C(c1cc(F)cc(F)c1)=O Cc1cc(F)cc(C)c1C(c1nnnn1C1CC(F)(F)C1)NCCc1nncs1 C#CC1CN(C(=O)C(c2ccc(C)o2)C)CCN1C(=O)CCc1ccc(Cl)cc1 c1(C(N(CCCNC(C(C)=CC)=O)C)=O)cc(OC)ccc1Cl C1(C)(CNC(C=C(CNC(c2cc(OCC)no2)=O)C)=O)CCN(C)C1 C#CC1(NC(=O)C(c2cnn(C)c2)NC(c2c[nH]cc2CC)=O)CCCOC1 N1(C(CCC(=O)NC)=O)C2CCCC1CN(C(=O)CC(C)(O)c1ccccc1)C2 c1(C(C)OC)nc(C)c(C(=O)NC(C2CCN(C(=O)C=NOC)C2)C)s1 c1(C(=O)NC2CC(NC(=O)CC3CCCO3)CC2O)cccc([N+](=O)[O-])c1Cl CCC(Cc1cnc[nH]1)C(=O)N(CC(C)N(C)C(C1CC(F)(F)C1)=O)C CCCC(O)C(=O)NCC1CC(NC(c2cc(SC(F)(F)F)c[nH]2)=O)C(O)C1 Cc1cc(C(=O)NCC2CC2CNC(c2nnc3ccccn23)=O)c(O)c(C)c1 c1(C(c2nnnn2C(C)(C)C)NCC2(C)CSC2)cn(-c2ccccc2)nn1 c1(C(N2CC(C(=O)OC)S2(=O)=O)=O)cccc2sc(-c3ccccc3)nc12 N1(C(C(C)N(C(C(C)=CC(C)(C)C)=O)C2CC2)=O)CCCCC1C C1(CC=C)(NC(=O)CCCC2CCCC2)CN(C(=O)CC2CCC2C)C1 C1(CC(=O)NC(CC)CN(C(=O)CCCc2ccccc2)C)CCCNC(=O)C1 Nc1cc(F)cc(F)c1C(=O)NCC1(O)CCCN(C(C2CCC2)=O)C1 N1(C(CCCSCC)=O)CC(C(=O)O)C1(C)C c1(C(=O)NC(C)CCCNC(C2CC3(C2)CC(F)C3)=O)cnn2ccccc12 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CC(NC(C(C)(F)F)=O)CC1O c1(C(=O)NCC2CCCCN2C(=O)C(O)C(F)(F)F)ccc(F)c(F)c1 C1(CNC(Cc2c(C)non2)=O)CCCCC1NC(C1CCCCN1C)=O c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)S(N)(=O)=O)ccc2ccnn2c1 CCCC(C)(O)CC(=O)N1CC(CNC(c2ccns2)=O)(COC)C1 C12(NC(C(C(C)C)OC)=O)CCC(NC(C3CC(F)(F)C3(F)F)=O)(CC1)C2 Cc1ccc(C=CC(=O)NC23CC(NC(=O)COc4cnn(C)c4)(C2)C3)nc1 N1(C(=O)NCCCn2cc(Br)nn2)CCCC1C1CCOCC1 N1(C(C(C)=O)=O)CC(NC(c2ncccn2)=O)CC(C)C1 N1(C(CSCC=C)=O)CCCCC12CN(C(c1cc(-c3ccccc3)co1)=O)C2 N1(C(CC(C)SC)=O)CC(NC(c2cnc(CO)nc2C)=O)CC(F)C1 c1(OCC(=O)NC2CCC(CNC(CC(C)(F)F)=O)C2)ccccc1C#N c1(C(C2CC(NC(CC3(OCCO)CCC3)=O)C2)=O)coc(C2CC2)n1.CCOC C1(CNC(C=C(C)C2CC2)=O)CCN(C(=O)Cc2n[nH]c(=N)s2)C1 C=CC(CC)CC(=O)NCCC1(NC(C2CC23CCCC3)=O)CCCC1 C1(C(=O)NCC(CC)(C)NC(=O)OC(C)(C)C)Cc2c[nH]cc2S1(=O)=O c1(OC(C)C)ccc(-c2cn(CCC(=O)NC(C)C(O)C(F)(F)F)nn2)c(Cl)c1 N1(C(CC2CC(=C)C2)=O)CCC(CCNC(c2cnc(CCC)s2)=O)C1 N1(C(=O)Nc2cc(C)nnc2C)Cc2cccc(Br)c2C1 c1(C(=O)NCC(N(C(CC(CC)O)=O)C)C2CC2)ccn2ccnc2n1 c1(C(=O)NCC2(CNC(C3C(C)C3)=O)CC2)csc2cc(Cl)ccc12 c1(C(=O)NC2CN(C(c3ncc(OC)cn3)=O)CC2F)cc(SC)ccc1OC C12(CNC(c3c(C(C)=O)cccc3)=O)CCCN(C(c3ccnc(C)c3)=O)C1C2 c1(C2CC(NC(C(CC)c3ccccc3)=O)C2)ccc(O)c(F)c1 c1(CC)cc(C2c3nnnn3C3(COC3)N2)ccn1.C1(COC)CCOC1 N1(C(N(C2C(C)CNCC2)C(c2cc(I)c(O)cc2O)=O)=O)CCC12CCCCC2 C1(C(=O)NC(c2cccnc2)C(=O)N2CCC2C2CC2)CC=CC(O)C1 c1(C(N2CCCN(C(CSCCOC)=O)CC2C)=O)cc2ccccc2cn1 N1(C(C(CN(C(CCSC)=O)C)C)=O)CCCC[Si](C)(C)C1 c1(CC(=O)N(CC(CC)NC(=O)C(F)Cc2ccccc2)C)ccc(O)nc1 C(=O)(C(CC(N)=O)NC(=O)CC#N)N1CC(C(=O)NC23CC(C)(C2)C3)OCC1 Cc1nn(C)c2c(N3CC4CC=CCC4C3)nc(=NC3CC4C(C3)C4(F)F)[nH]c12 c1(-n2cc(C(CC)NCCNC(C(C=C)OC)=O)nn2)ccc(Cl)cc1 c1(C(N2CC3C(C(=O)NC(CC)C(N)=O)(C3)C2)=O)ccc(C(F)(F)F)c([N+](=O)[O-])c1 C(CN=C(NCc1ccc(C)cc1)NCC(F)C(=O)N(C)C)OC Cc1ncc(C(N2CCC(CO)C(NC(=O)Cc3cnnn3C)C2)=O)c(C)n1 C1(N(CC(C)NC(=O)CC(O)c2ccccc2)C)CCCN(C(C)(C)C)C1=O CS(=O)(=O)c1ccc(C(N2CC3CC2CS3)C(=O)NCc2ccccc2Br)o1 C1(CNC(CNC(CC)=O)=O)CN(C(=O)CCC2CCCCC2)C(C)(C)C1 n1(CC)ncnc1C(C)NC(C12CC(NC(C3CCC(C)O3)=O)(C1)C2)=O N1(C(c2c(OC)oc(C)n2)=O)CCN(C(C2CC2C(F)F)=O)C(C)C1 Cc1cc(NC(C2CC3CC3N2C(C2CCC(O)CC2)=O)=O)cc(Br)c1C Cn1ccnc1C(=O)NCCc1ocnc1CNC(C1CCC1F)=O C(=O)(C(CC)C(C)C)N1C(CCNC(C2(CC#C)CCCO2)=O)CCC1 c1(OC)nsc(OC)c1C(N1CCC(C(C)NC(=O)C(=O)NC2CC2)C1)=O C(CC1=CCN(C(=O)C(F)CC2CCC2)CC1)NC(C1Cc2nccnc2C1)=O N1(C(c2c(CC)[nH]cc2)=O)CCOCCC1C(=O)NCCn1nncc1C C(C1=CCN(C(=O)CCc2ccnc(Cl)c2)CC1)NC(c1ccc(CO)s1)=O C1(CN(C(C2(CC)CCC2)=O)CC)CCN(C(c2cc(Br)co2)=O)CC1 C1(OC)CC2(C1)CC(C(=O)NCCC1CCN(C(=O)C(C)=CC3CC3)C(C)C1)C2 C1(CC(N2C(Cc3cn(CCOCC)nn3)CCC2)=O)CC2(CCC2)C1 C=C(C)C(O)CC(=O)NC(C)CNC(=O)Cc1cccnc1Br c1(C(c2cn[nH]c2)NC(c2cnco2)C)nnnn1Cc1ccco1 N12CCCC(C(F)F)(C1)OC(=O)c1ccc(cn1)C2=O.C(C)(C)(C)OC(C)C c1(C(N(CCCCNC(C2(C)CC2)=O)C)=O)cc(C(F)(F)F)cc(F)c1 c1(NC(CCN(C2CC3CCC2N3)CC)=O)cccc([N+](=O)[O-])c1 c1(CCC(=O)NCCC(C)(C)NC(C(COCC)C)=O)ccc2c(c1)COCC2 C1(F)(CNC(=O)CCC2CCCO2)CCN(C(C2CCC(=O)NC2)=O)CC1 N1(C(=O)OC(C)(C)C)CC(C)(C)C(C(=O)NCCN2CCSCC2)C(C)(C)C1 C1(NC(C(C)OCC(F)(F)F)=O)CCCCC1CNC(=O)CC1CC(C)(C)C1 Cc1csc(Cl)c1C(N1CCOC(CNC(=O)Cn2cnc(C#N)n2)C1)=O C1(C(NOCC=C)=O)CCN(C(=O)C(C)CC(F)(F)F)C(C)(C)C1 N1(C(CCCCCC=CC)=O)CCC2(CCC(OCC)C2)C1 C(=O)(C1Cc2ccc(F)cc21)NC1(C2CCN(C(c3csc(C)c3N)=O)C2)CC1 c1(N2CCN(CCOC)CC2)nc2ccc(Cl)cc2c(=NC(C)C2CCCCO2)[nH]1 N1(C(c2n(CCC)ccc2)=O)CC(N(C)C(C2CC23CCCC3)=O)C2(CC2)C1 CCCC(CNC(c1cnn(CCO)c1C)=O)C(=O)NC1(C(N)=O)CCCOC1 Cc1ccc(C=CC(=O)NC(C)CN(C)C(c2cc(C)c(Cl)s2)=O)cn1 c1(C(=O)NCCC2CCN(C(CC(=O)OC)=O)C2)ccc(S(=O)(=O)C(F)F)cc1 c1(NC(=O)NCC2(SC)CC(O)C2)ccc(-c2ccccc2)c(F)c1 c1(C(N(C2CCN(C(C3C=CCS3)=O)C2)CC2CC2)=O)cnc(O)c(F)c1 c1(C(C)C)ccc(C=CCC(=O)NCC2CC2NC(C2(C)CC=CC2)=O)cc1 N1(C(COC)=O)CCCC(NC(=O)C=Cc2nnc(C(C)C)o2)C(F)C1 c12ccc(c(Cl)c1)OCCN(C=O)C2.CC1CCN(C(=O)N(C)C)CC1 N1(C(C2C(C=C)OCC2)=O)CCCN(C(=O)Cn2cc(C(C)=O)nn2)CC1C c1(CN2CC(NC(c3ccncc3C(F)(F)F)=O)C2)cc(F)c(F)cc1Br C12CCN(CC1)C13CC(C1)(C3)NC(=O)NC2.O=C(C(O)CC1CCCCC1)O.CCO C(CC(=O)N(C1CC(C(=O)NC)C1)C)(C(C)CC)NC(C(C)OCCOC)=O CC1CC2CN(C(=O)C(=O)NC3COCC3N3CCOCC3)CCN2C1 C1(C(N2CC3C(CNC(CCCOCC)=O)C3C2)=O)CSC(c2ccccc2)=N1 c1(NC(=O)NC2CCC(NC(c3cccnn3)=O)C2)ccccc1Cl c1(C(=O)NCc2ncc(C(=O)NCCC3CCN(C)C3)cn2)cc(F)cc(F)c1 CC(C)CCCCC(=O)NCCN1CCCN(C(C23CCOC2CC3)=O)CC1 C1(C(=O)NC(C)CCNC(c2cnc(O)n2C)=O)CCc2nc[nH]c2C1 N1(C(C2CCC(C(=O)OC)CC2)=O)CCC(NC(=O)CCCC(N)=O)C(F)C1 C1(C(=O)NCC(CNC(=O)CCc2ccco2)OC)CCC2(CC2)C1 Cc1ccc(F)c(C(=O)NC2CN(C(c3ccc(OCF)cc3)=O)CCC2C)c1 C1(C(N(C2CC3C=CC2C3)C)=O)CC1C1CN(C(=O)CCCCC2CC2)C1 N1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCC2(CC1)OCCO2 c1(OC)cc(Cl)ccc1C(N1CC(NC(c2c[nH]nc2C)=O)C2CC2C1)=O C1(CC(=O)NCC(C)N(C(c2cnc(C(C)C)[nH]2)=O)C)CCN(CCF)CC1 C(CCS(N)(=O)=O)(C(=O)O)n1cc(-c2ccc(OC)nn2)nn1 C(=O)(C(F)CCC(C)(C)C)NCC1C(NC(C(C)(C)OCCC)=O)C1 N1(C(CC2N(C(C3(CC=C)CCOC3)=O)CC3(CC3)C2)=O)CC2COCC(C2)C1 C1(C(N2C(C)(CC(=O)NCc3c(CC)onc3C)CC2)=O)CC12CCOCC2 Cc1cc(Cl)c(C(=O)NC2CC(CNC(C3CCO3)=O)C2)c(Br)c1 C1(NC(C(C(C)O)C)=O)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)CCC1(C)C C#CCC(C(=O)N1CCC(CN(C(=O)CCn2c(C)csc2=O)C)C1)C1CC1 N1(C(C2C(C)COCC2)=O)CC(C)N(C(c2ncn3c2CCC3)=O)C(C)C1 C=C(Cl)CCC(=O)NCCC1CN(C(c2ccc(SCC)cn2)=O)CCO1 c1(C(=O)NC(CC(C)NC(C=Cc2c(C)noc2C)=O)C)noc2ccccc12 c1(CN(C(=O)CN(C2CC(C#N)C2)C(C2CC2Cl)=O)C)cc(F)ccc1O CCCCC(C(=O)NC1CC(C)(NC(c2[nH]nnc2C)=O)C1)C(C)C N12CCC=C(C(=O)Nc3cc(ccn3)C1)C2.Cc1ncc(Br)c(C(=O)N(C)C)n1 CN1CCC(CC(=O)NCc2cc(C(N3CC(CO)C3(C)C)=O)co2)C1=O C1(C(=O)O)COCCN(CC2CCC(F)(F)CC2)C1 c1(C(N2C(CCNC(CSCC#C)=O)COCC2)=O)ccnn2ccnc12 c1(C(N2CC(CNC(=O)CCCCF)C2)=O)nc2ncccn2n1 c1(C(C)C)cccc(C(=O)NCC2(C)CCN(C(=O)CC3CC3C)C2)n1 C(=O)(CC(C)CF)NC(C1CCCC1)CNC(C=C(C)C(C)(C)C)=O c1(NC)cc(C(=O)NCC(C2CCC2)NC(=O)C=CSC)cc(Cl)n1 c1(CCC)noc2nc(C3CC3)cc(C(N3CCCC(C)(C)C3CO)=O)c12 C1(CC)CN(C(C2CC(C)CN2C(c2cnc(C)nc2)=O)=O)CCO1 N1(C(c2ncn(CC)n2)=O)CC(C(=O)NC2CC(O)C(F)C2)OC(C)C1 C(C(CC)CCC)(c1nnnn1CC1CC1)N.c1(NC)ncc(CC2CCCO2)[nH]1 C(CCC(C(=O)NC1(c2nc[nH]n2)CC1)NC(=O)CCCCC#N)OC C(=O)(C(C)C(C)(C)C)NCC(C)N(C)C(c1ccc(C(=O)OC(C)(C)C)o1)=O C(C(=O)N1OC2CCC1C2)N(C(C1CC1F)=O)CC1CC1 C1(NC(Cc2cn(CC)nc2)=O)CN(C(=O)C=C(Cl)Cl)C2(CCCCC2)C1 c1(OC)ccc(NC(=O)CN(CC(C)C)C(=O)Cn2cc(Cl)cn2)cc1 N1(C(C(C)NC(=O)CC2=CCCC2)=O)CCC2(CC=CCO2)C1 c1(C(=O)NCC(CC)NC2CC2)cccc(C(C2CCC2c2nncn2C)=O)c1 c1(CC)c(C(N2CCOC(C(C)NC(c3cocc3C)=O)C2)=O)ccn1C C1(C(N2C(C)C(c3ccccc3)CC2)=O)CCC(F)(F)C1O C1(C(N(CC(C)N(C(c2n(CC=C)ccc2)=O)C)C)=O)C(F)(F)C12CCC2 C(C)(C)(C(C)CC(=O)NCc1ccc(C)o1)NC(c1c(CC)noc1)=O CCCCCCCCC(=O)NC1CC2CCC1CC2NC(=O)C(=O)NC1CC1 CCCC(CC(C)C)C(=O)NC1(COC)CCN(C(=O)C=Cc2cn[nH]c2)CC1 C1(C(N(CCCN(C(CNS(CC)(=O)=O)=O)C)C)=O)CCCCN1C c1(NC)c(C(N2CCCC2CNC(C2CCN(C)C2)=O)=O)sc2nccnc12 CC(C)C(C)(CNC(=O)CCc1ccnn1C)NC(=O)CCC1CCCC(O)C1 c1(C(N2CCC(Cc3ccccc3)(OC)C2)C(=O)NCCC)ccc(Br)cc1Cl N1(C(c2c(CC)nns2)=O)CC(C(=O)N(CC(C)(C)O)C2CC2)CC1(C)C C(c1cccnc1)=C(C)C(=O)NCC1(OC)CCN(C(=O)C=Cc2sccc2C)C1 Cc1ccc(N)c(C(=O)NCCC2CCCN(C(=O)CCc3cc[nH]n3)C2)c1O C1(C(=O)NC2C(C)(C)CN(C(=O)CCCn3cccn3)C2)CCCCC1C1CC1 C(c1ccc(C)s1)=CC(N1CCC(N(C(c2csc(C(C)(F)F)n2)=O)CC)C1)=O c1(C(N2C(CNC(C3CCS(=O)(=O)N3)=O)CC(O)C2)=O)cc2n(n1)CCCN2 N1(C(CC2(COC)CCCC2)=O)CC2CCC(C1)C2NC(=O)C1=CCCCC1 c1(C(=O)NC2CC(C)N(C(=O)CC3CCC(F)(F)C3)CC2)ccnc2[nH]nnc12 C1(CNC(C2CN(C)C2)=O)CC2(CO1)CN(C(=O)C(C)(C)c1ccccc1)C2 N1(CCC)CCCC(C(N2CC(N(C)C(c3cc(CC)on3)=O)C2)=O)C1 c1(C(=O)NCC2CC3CCC2N3C(=O)CC2=CCCCC2)ccc2c(c1)OCO2 CC(C)CC(C)CNC(=O)C(C)(CO)NC(=O)C(C)Cn1cccn1 c1(NC)snc(C)c1C(=O)NCCN(C(=O)C(C)O)CC1CC1 c1(CN=c2nc(CCC)[nH]s2)ccc2c(c1)CN(C(c1nc(=O)n(C)[nH]1)=O)C2 C1(CNC(C(C(C)C)N(C)C)=O)CN(C(c2nnn(C)c2N)=O)CCC1(C)C c1(C(=O)NC2CC3(C(NC(CCCCC=CC)=O)C3)C2)cc(C)c(Cl)c(C)c1 c1(SC)ccc(CCC(=O)NC2CC23CC(NC(c2cc[nH]n2)=O)C3)cc1 c12nc(oc1C)CN1CCC1C(=O)N2.c1(C(=O)OCC)cc(C(C)C)[nH]n1.C Cc1c(C(=O)NC23CCCC2CN(C(=O)C(C)(F)F)C3)cccc1S(N)(=O)=O N1(C(CCC(C)C)=O)CCN2C(=O)C(NC(=O)CNS(=O)(=O)C(F)(F)F)CC2C1 C(=O)(C=CS(F)(F)(F)(F)F)NCC1CCCN(C(c2ccc(C#N)s2)=O)C1 N1(C(NON(CC(=O)NN)C)=O)CCC(NS(C)(=O)=O)CC1.C1(C)CC1 C1(C(=O)NCC2CC2)CC2(CCN1C(c1cccc[n+]1[O-])=O)CC2 c1(C(=O)NCC(C)NC(CC(CC)C(F)F)=O)cc2cccnc2cn1 C(CNC(C1CCC(F)(F)C1)=O)(CC(F)(F)F)NC(CNC(CNC(C)=O)=O)=O c1(C(=O)NC2CC(CNC(c3c(C)nn[nH]3)=O)C2)ccc2cnnc(O)c2c1 CCCC(CCC)S(=O)(=O)CC1CC(C)N(C)C1 c1(CC(=O)N(C(C)CCNC(c2cc(F)c[nH]2)=O)C)ccc(N)cc1 C1(CNC(COCCCC)=O)CCCCN(C(=O)Cc2cccc(C(N)=O)c2)C1 C12(NC(c3cc(OC)n(C)n3)=O)CCOCC1CN(C(=O)Cn1cncn1)C2 CC(CN=c1[nH]c(N2CCc3ncncc3C2)nc2c1SCC2)C(F)F CC1CN(C)C(C)CC1NC(c1n[nH]cc1CNC(C1CC2(C1)CC21CC1)=O)=O c1(C(C)NC(=O)OC)ccc(NCCN2CCCCC2C)c([N+](=O)[O-])c1 C(C(=O)NCC(C)NC(c1nc(-c2ccco2)oc1C)=O)(C(C)C)OC c1(C(N2CCC(CNC(C(CC#C)C3CC3)=O)C2)=O)ccc2nccn2c1 c1(OC)cc(C(C)NCc2ccnn2C2CC2(F)F)c(F)cc1F c1(C(=O)NC(CSC)(C)C(=O)NCc2ccn(C3CC3)n2)cc(C)nnc1C CCS(=O)(=O)CCNC(C1(F)CCN(C(=O)C(F)CC2CCOC2)C1)=O N1(C(C23CC(NC(CCCC4C(C)C4)=O)(C2)C3)=O)CCC(CC2CC2)CC1 C1(NC(=O)CC2CC2(Cl)Cl)CC2CN(C(c3[nH]cc4c3CCCC4)=O)CC2C1 c1(C(=O)NC2CC(C)N(C(=O)C3=COCCC3)CC2)ccc2c(c1)OC(C)(C)O2 C1(C(N(CCC(=O)NCCN2CCCNC2=O)C(C)C)=O)CCC(C)(O)CC1 c1(CC(=O)N(CC(C)CNC(C2(CF)CC2)=O)C)ccnc(C(F)(F)F)c1 C1(C(=O)NCCn2cc(C(=O)NC(C)Cc3cn[nH]c3)nn2)(CF)CCOCC1 Cc1ccc(NC(C2CC(F)(F)CN2C(c2cnccc2C)=O)=O)c(Br)n1 CC(C)C(C(=O)NCC1CN(C(=O)CSC(C)C)CCO1)NC=O C(C1=CCCCCCC1)(c1nnnn1CCCF)NCc1cnc(C)o1 CCCC(CC)C(=O)N1CCC(O)(CCNC(=O)CCc2cnc(C)s2)CC1 N1(C(c2ccnc(F)c2F)=O)CC2CN(C(c3c(Cl)nsc3Cl)=O)CC2C1 C1(=CCNC(CC=C=C)=O)CCN(C(=O)CSCC2CCCO2)CC1 C1(NC(C2(C)COC2)=O)CN(C(C2(c3ccc(Cl)c(Cl)c3)CC2)=O)CC12COC2 C1(CC)C(C(=O)NCCN(C)OC)CCN1C(c1cccnc1)=O c1(OC)cccc(CO)c1NC(=O)C(N1CCC(OC)C(O)C1)=O C(=O)(C(O)C1=CCCCC1)NCC(CC)(C)NC(c1c(C)ncn1O)=O C(c1ccc(F)c(C)c1)=CC(=O)NCC1N(C(COCC#C)=O)CC(O)C1 Cc1cc(O)cc(C)c1CCC(=O)NCCNC(c1ccc(SC(F)(F)F)o1)=O C1(COC)(NC(=O)C=NOC)CCCN(C(c2sncc2Br)=O)C1 C(CCCC(=O)NC(C)CNC(c1ccc(-n2cncn2)cc1)=O)SC c1(CC)cc(C(=O)NC2CC(CNC(=O)C(C(C)C)NC(N)=O)C2)cc(F)c1 c1(C(=O)NC(CNC(c2cscc2C2CC2)=O)C2CC2)cc[nH]c2nccc1-2 C1(NC(c2n(C)c(S)nn2)=O)CCSC12CN(C(C1CCCC13CCC3)=O)C2 C1(C(C)C)CN(C(=O)CCOC2CC2)CCN1C(C1(C)CCCCO1)=O C1(COC)CN(C(C)=O)CCN1C(c1snnc1C)=O.C12CCCCN1C(=O)C2 C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(=O)CCN2CCCCC2=O)CC1F C1(CNC(C(CC)SC)=O)CC2CC2N1C(c1cccc(CO)n1)=O c1(CN(CCCC(=O)OC)CC)cnoc1C(=O)NC c12c(F)cc(F)c-1c2F.Brc1ccc(CNc2ccncc2)o1 C1(CNC(c2c(OCC)n[nH]c2)=O)CC2CCC1N(C(=O)Cc1nc[nH]n1)C2 C1(NC(=O)C(C2CCC2)NC(C2CCC(CO)CC2)=O)COC2(CCC2)C1 N1(C(C(N2CC(NC(=O)C(F)(F)F)CC(C)C2)=O)=O)CC2(C1)CS(=O)(=O)C2 c1(CC(C)OC(CCOC)=O)ccc(F)c(OCC)c1F c1(C(N2CCN(CC(C)(C)NC(CC(=C)C)=O)CC2)=O)cc2c(Cl)cccn2n1 C(=O)(CCC(=O)N(C(C)CN(C)C(c1cscc1Cl)=O)C)N(CC)CC Cc1nn(C)cc1S(=O)(=O)NC1CC(C(=O)Nc2ncc(Cl)cc2Br)C1 C1(C(N(C2CCN(C(=O)CC(C)C3CCCC3)CC2)CCC)=O)CCOC1(C)C c1(OC)cc(C(N2CC3CC2C3NC(=O)Cc2cc[nH]n2)=O)ccc1Br C1(C=O)(CCl)CN(C(=O)C(C2CCCOC2)NC(C=CC)=O)C1 c1(C(N2CC(C(=O)Nc3c(C)ccc(F)c3)C2)=O)cc(C)c2cc[nH]c2c1 C12(CCNC(COCc3c(C)ncs3)=O)CCC1CN(C(c1ccccn1)=O)C2 c1(C(N2C(CC(=O)NCc3ccco3)CCC2)=O)ccc2nn[nH]c2c1 C1(CNC(C(CCC)OCC)=O)CCC2(CCC2)CN1C(C1CCSCC1)=O N1(C(=O)COc2cccc(F)c2)CC23CCCC2(C1)CN(C(C1CCSC1)=O)C3 C(=O)(C1=CCC(C)CC1)NCCC(CNC(c1nccc(C#C)c1)=O)O c1(CN2C(C(N3CCOC(c4ccccc4)C3)=O)CCCC2)ccc(O)c(Br)c1 CC1CC(CO)(NC(=O)C(C2(O)CN(C(=O)C=CC(C)(C)C)C2)F)C1 c1(N)nnc(O)c2ccccc12.Cc1cnc(CCO)cn1.n12nnnc1N1CCC2C1 C(=O)(C(C)C(O)CCCC)NCc1c(C(N2CCC(C#C)C2)=O)n[nH]c1 CC1(C)C2CCC1(CC(=O)NCCCC1CCCN1C(=O)C=CI)CC2 N1(C(C=C(CC)C)=O)CCC(CNC(=O)CCCOC)C12CC2 c1(OC)cc(C)ccc1NC(=O)NC1CCN(C(C2CCC3(CC3)C2)=O)C1 c1(C(N(C2CCCC2C#N)C)=O)cnn2c(-c3cc(F)ccc3F)ccnc12 CC1CC2CN1C2=O.c1(CN(C(=O)CSCC(N)=O)C)ncn(C)n1 c1(C(=O)NC(c2ccc(C#N)s2)C)n[nH]c2c1CCN(C(=O)CCCC1CC1)C2 C(=O)(CC1=CCOCC1)N1CCN(C(Cn2nnc(C(C)(C)C)n2)=O)C(CO)C1 C1(NC(CNS(NC)(=O)=O)=O)CCC(NC(c2cnoc2C2CC2)=O)CC1 c1(C(N(CC(O)CNC(C2CC2C(C)(F)F)=O)C)=O)cccn1CC1CC1 C1(NC(C=COCC)=O)CC2CC(NC(C3CCC4(CCC4)O3)=O)C1C2 C1(C(N)=O)CCCCCN1C(=O)Cc1ncn2c1CCC2 CCC(CC(=O)N(C1CCCN(C(=O)CCCNC(N)=O)C1)CC)C(F)F C1(NC(=O)NCCSC(F)(F)F)CC(=O)N(c2cccc(Br)c2)C1 Cn1cc([N+](=O)[O-])cc1C(=O)NC1CC(NC(C2CC3CCC2CCC(=O)N3)=O)C1 c1(C(=O)NC23CCCN(C(CCNC(=O)NC)=O)C2C3)cc2n(n1)CCOC2 Cc1cc(CNc2ccsc2C(=O)NCc2ccncc2O)cc(C)c1 Cc1onc(C(N2CC(NC(c3cnoc3-c3ccccc3)=O)C2)=O)c1[N+](=O)[O-] CC(C)C(C(=O)NC1CCC(NC(=O)C(C)(C)CN(C)C)CC1)N(C)C C(=O)(C(C(C)(C)C)NC(=O)C(C)S(C)(=O)=O)NCCc1ccc(C)nc1 N1(C(C2(C#N)CC2)=O)C(CNC(c2cc(C3CC3)nnc2O)=O)CC2COCC12 N1(C(C(C)Cc2ccccc2Cl)=O)CCCN(C(=O)CCC2CC2)C(CO)C1 c1(CCC(=O)OC(C)(C)C)ccc(Br)cc1C.C1C(CO)CNC(=O)N1C N#CC1(C(=O)NCCSC2CC(F)C2)CC1 N1(C(C)=O)CCC(C)C1C(=O)NCCF C1(NC(=O)Cc2cc[nH]n2)CC2CC1N(C(c1cc(NC3CC3)ncc1Cl)=O)C2 CCC(CC(=O)N1CCCC(CCC(=O)NC(c2c(C)n[nH]c2C)C)C1)C(F)F c1(C2(C(=O)NCC3CN(C(C4CC(F)(COCC)C4)=O)C3)CC2)ccc(O)nc1 N1(C(c2cccc(CC)c2)=O)CC2(CCCN2C(c2cc(Cl)c(Br)s2)=O)C1 C(=O)(C(C)(C)CCCF)N1CC(C)N(C(c2ccncc2)=O)CC1 C1(NC(C2C(C)CCOC2)=O)CC=C(C(=O)NCc2nc(C(C)C)n[nH]2)C1 N1(C(CSc2n(C)c(Cl)cn2)=O)CC(C)(C)CC1CNC(C1(C#N)CCCOC1)=O C1(C)(NC(CCC=C(C)C)=O)CCN(C(=O)Cn2nc(O)ccc2=O)CC1 C(=O)(CCCC(F)(F)CO)N1C(CNC(=O)CC2CCC(=O)O2)CC2(CC2)C1 N1(C(C(CC)COC)=O)CC(C)(C)OC2(C1)CN(C(C1(Cl)C3CCC(=O)C13)=O)C2 Cc1ccc(F)c2c1N(CCc1ccnn1C1CC1)CCC2 c1(C(C(=O)OC2(C)CC2)NC(C2(O)CCOC2)=O)cn(CC2CCCO2)nn1 c1(COC(C2(c3c(Cl)cccc3Cl)CC2)=O)cc2cccc(Br)c2[nH]1 Cc1sccc1C(=O)NCCc1cn(Cc2occc2C(=O)O)nn1 Cc1c(C(=O)NCC(C)N(C(=O)CC(C)NC(N)=O)C)[nH]c2c(Cl)cccc12 c1(C(C(N2CC(COC)(NC(=O)CC(C)CF)C2)=O)O)ccc(OC)cc1 Nc1ccc(C(=O)NCC=CCNC(c2cn(C3CCC3)nn2)=O)nc1N C1(C(=O)NCCCN(C(=O)C(C)C2CC2)CC)CCCCC1O.S(=O)(=O)(CC)N N1(C(CC(C)CNC(c2cncc(O)c2)=O)=O)CC(C)C(N=[N+]=[N-])C1 n1(CC(=O)NC2CC(NC(C(CC3CC3)OC)=O)C2)nnc2ccccc12 Cc1ccc(C(C)NC(C2CCCN2C(c2scnc2Cl)=O)=O)cc1 C1(CNC(=O)CC2CC3CCC2C3)(CO)CCN(C(C2CC(O)C2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCCCC1CN(C(=O)Cc1occc1C)C c1(C(=O)NCCNC(C2CC(N(C)CC)C2)=O)cnc(S)[nH]1 C(CCC(=O)NC(Cc1cnc[nH]1)CO)N(C)C.C12(CC1(C)C)C(=O)N2 c1(NCCCCNC(c2c(C)nco2)=O)ncccc1C#N Cc1nc(CO)ncc1NC(C1CCCC1CNC(C1(C)CC1(C)C)=O)=O C(=O)(N=c1[nH][nH]c2ccccc12)C1C(C(=O)Nc2nccc(F)c2F)C1 c1(C(=O)NCC(CC=C)NC(c2cnn(C)c2COC)=O)cc(C#N)cn1C Cc1ncn(O)c1C(=O)NCC1CCC(NC(c2cn(C3COC3)nn2)=O)CC1 N1(C(Cn2c(C)cc(C)nc2=O)=O)CCCC2CCN(C(=O)C(F)F)CC12 C1(C(N2CCC(CCCCNC(c3c[nH]c(=N)o3)=O)CC2)=O)CC12CCSCC2 N1(C(=O)CC2(C)CC2(F)Cl)CCC(O)C(C(=O)NCc2n(C(C)C)cnn2)C1 N(C(=NCCC1CCCC1)NCc1ccsc1)C(c1cccc(F)c1)C C(CCC(C)C(=O)NC1CN(C(=O)CCN2CCC2)CC1c1cncn1C)OC C(C)(CCCCNC(=O)CCC1CC1(Cl)Cl)NC(C(C)C)=O c1(C(CNC(C(F)=CC)=O)NC(c2scnc2Cl)=O)ccc(F)cc1F C(C(=O)NNC(=O)Cc1ccccc1F)n1ncc(C)c1CC(C)C C1(C(=O)N)CC(F)CN(CC2(C(=O)OC)CC2)C1.c1(S)ccc(F)c(C2CC2)c1 CCC(C)(CC)C(=O)N1C2CCC1C(CNC(c1cn3c(n1)CCC3)=O)C2 c1(OC)ccc(C(N2CCC(C(C)NC(=O)Cc3ccnn3C)CC2)=O)c(Cl)n1 C(=O)(CC(CN(C)C)C(F)(F)F)NC(CCOC)CNC(c1ccn(CC)n1)=O CC1CN(c2cc(NCCOc3ccc(F)cc3)ncn2)CCCO1.C1CS1 CC1CC(N=c2[nH]c(=NCCc3cccc(F)c3F)[nH]c3ccsc23)CCO1 c1(N(C)C)ccc(C(c2nnnn2CC2CCCO2)NCC23CCCC2C3)cn1 c1(C(=O)NC2CCC(N(C(c3cnc(C)s3)=O)C)C2)cccc(N(C)C)n1 N#Cc1c[nH]c(=NC(=O)C23CC(NC(c4cc5c(s4)CSC5)=O)(C2)C3)cc1F c1(-c2ccc(C(N(C)C)=O)cc2)cnc2c(C(N3CCC(O)C3)=O)cccn12 CC1CN(C(=O)NCCCl)CCC1N=c1ccc(Br)c(S(=O)(=O)N2CCCC2)[nH]1 N1(C(C(COC)OC)=O)CC2(C1)CN(C(c1nn(C)c(C)c1Cl)=O)CC2CO C1(CC#C)CCCCN1C(=O)COCCN(C(=O)COCC(=C)C)C Cc1cc(C)c(C(N2CCCCC2CC(N)=O)=O)cn1.C12CCCC(C1)C(=O)N2 Cc1ncnc(O)c1CCC(=O)NCCCC(C)(C)NC(c1cnsc1)=O c1(C(N(C(c2onc(C)n2)C)C)=O)cccc(Cl)c1C(F)(F)F Cc1nc(CCC(=O)NCCC2CN(C(C3COC(=O)N3)=O)CCO2)oc1C N1(C(C(CSC)C)=O)CCCC2CN(C(=O)Cc3c[nH]c4cnccc34)CCC12 N1(C(C2CCC(C)C2)=O)CCN(C(=O)C(C)(C)n2cccn2)CC(O)C1 c1(C(=O)NCC2(NC(=O)Cc3ccsn3)CCOC2)noc2c1CCCC2 c1(NC(=O)CC2CCCN2C(=O)C(O)CC2CC2)ccc(O)nc1 N1(C(CCc2ccc(C#C)cc2)=O)CC2COCCC2(NC(=O)CCC(N)=O)C1 N1(C(c2ccc(OCC)nc2)=O)CC2(CCC2)CC1CNC(=O)C(C)S(C)(=O)=O c1(OCC(=O)NC(CC(C)NC(Cc2c(C)nc(C)s2)=O)C)cccc(Cl)c1C c1(C(N2CCN(C(CC3CCCC(C)C3)=O)C3(C2)CC3)=O)cnc2c(c1)CCOC2 C123CC(CN(C1)C(=O)C(=O)N2)C3.c1(SC)cc(C)nc(OC)n1 CC1(CCNC(C2C3CCC2CC3)=O)CCN(C(c2cncs2)=O)CC1 C1(C(=O)NC(C)CC2CN(c3ncc(C4CC4)cn3)C2)CCS(=O)(=O)C1(C)C CC1=NN(C)C(=O)C1CC(=O)N(C(CNC(C1(O)CCOC1)=O)C1CC1)C c1(C(N(CCOC(C)C)CCSc2ccccc2)=O)cc(-c2ccn(C)n2)on1 c1(C(N2CCC(NC(C(CC)OC)=O)C2C)=O)nc(C(F)(F)F)cc(C)n1 N1(C(C=C(C)CCc2ccccc2)=O)CCC(NC(C2(S(N)(=O)=O)CC2)=O)CC1C CCC(CC(C)C)C(=O)NCc1nc(CNC(=O)CC2CC(OC)C2)cc(O)n1 C#CCCCCCC(C(=O)NC1CCOC1)N(CCS(C)(=O)=O)C c1(C(=O)NC2CCC(NC(CC=CC=C)=O)CC2)cnc2sc(C)cn12 N1(C(c2nc(C)nn2C)=O)CCC(NC(C2CC23CCCC3)=O)CC1C Cc1cc(=NCC#CCCO)[nH]cc1S(=O)(=O)NCc1cn(C)nc1C(F)(F)F c1(NC(C2N(Cc3ccc(OC)cc3)CC(O)C2)=O)nc2ccccc2s1 C(C)(CO)(C(=O)N1CCCCC1CCCO)NC(C(CO)OC)=O C1(CCNC(C2CC=CCN2C(=O)CC2CC3(CCC3)C2)=O)CC2C=CC1C2 C12(C(=O)Nc3cccc(CNC(c4c(C)cccc4)=O)c3)CCC(C1)C2(C)C c1(C(=O)NCC2CCCC(NC(c3cnn(C)n3)=O)C2)cccc2ncnn12 c1(NC(CN(C(C)CO)C(C)=O)=O)cccc(C)c1C c1(C(c2n(CC=C)nnn2)NCc2csc(C(F)F)c2)ccccc1C(C)OC N1(C(c2c(C)noc2N)=O)CCC12CN(C(c1cnnn1-c1ccccc1)=O)C2 C1(C)(NC(CC=CCC)=O)CCN(C(=O)CC)CC1.C12CCCN(C1)C2=O C1(CCNC(c2nnc(C(C)(C)C)s2)=O)CCCN(C(C2C3CCC23)=O)C1 C=C(C)CCCC(=O)N(C)CCN1CCN(C(c2n[nH]cc2C2CCC2)=O)CC1 N1(C(C2CC(C(F)F)(OC)C2)=O)CCC2CN(C(c3ccnnc3)=O)CCC2C1 Cc1cccc(Br)c1C(N1CC(C(C)NC(=O)C(C)O)C1)=O C(C(C(=O)NC1CC2(CCC2)C1O)C(C)(C)C)NC(C(C)(C)n1ccnn1)=O c1(CN2CC(c3c(C)ccc(C)c3)OCC2C)cnn2cccc(C)c12 CCC(CNC(C1(NC(=O)Cc2cnns2)CCC1)=O)CC(C)C N1(C(C)(C)C)CCCC(C)(C(N2CCC(CCN3CCOC3=O)CC2)=O)S1(=O)=O C1(NC(CC(C=C)C)=O)CCOC12CCN(C(c1cc(C)c(Cl)s1)=O)CC2 Cc1ccc(C(=O)NCC2CCCN2C(C2(CO)CCCCO2)=O)cn1 c1(C(N2CCCC(CCC)(NC(=O)C3CC3)C2)=O)ccc(N)c(C)c1Cl c1(C(=O)NCC2N(C(CN3CCN(C)CC3)=O)CCC2)cc2cccn2cn1 C1(CNC(C(C2CC2)SC)=O)CCN(C(C2C=CCC2)=O)C1(C)C C(CC(C)CC)(C(=O)NCC(C)C(C)O)NC(c1nc(CCC)oc1)=O Cc1noc(CN2CCC(C(O)C(=O)O)CC2)c1C C(C(CC(F)(F)F)NC(c1cn(CC2CCCO2)nn1)=O)NC(CN(C)CC)=O c1(N(C)CCN2CCCC2)nc(=NCCSC(F)(F)F)[nH]c2c1CCC2 C(CC(C(C)(C)C)NC(=O)C(=O)NC1CC1)N(C(c1cc(C(CC)C)no1)=O)C C(c1cccc(F)c1)=CC(=O)NC(C(N1C(C(=O)OCC)CC(F)C1)=O)CN(C)C c1(NCC2C(CC(c3ccccc3)O)C2)c([N+](=O)[O-])ccc(F)c1F C(CC(C)(C)C)(C(=O)NCC1(O)CN(C(=O)CC2CCCOCC2)C1)OC c1(C(=O)NC(C)C(C)NC(c2sc(F)cc2Br)=O)cc2cccnn2n1 C1(C(=O)NC(CC)C(=O)Oc2ccccc2)CC(OC)CN1C(=O)C(CO)OC C(=O)(C1=CCC(C)CC1)N1CCC(C#C)(C(N2CCC(C(=O)OC)C2)=O)C1 N1(C(C(C)OC)=O)CC(C2CN(C(c3c(O)cccc3Cl)=O)C2)C1 C#Cc1ccc(C(N2CC(CNC(=O)CCNS(=O)(=O)CC)CCC2C)=O)cc1 C(=O)(C1=NOC2(CCC2)C1)N1CCC2(C(N(CCCF)CC)=O)C(CC1)C2 N1(S(CCC)(=O)=O)CCC2(CCCN(Cc3c(F)ccc(C)c3F)C2)C1 N1(C(C2C(C(=O)OCC)C2)=O)CCC(C)(c2cccc(Br)c2)CC1 c1(OC)cccc(-n2nnnc2C(c2cnn(CCO)c2)NCCCCCF)c1 Cc1cc(C(=O)N(C)CCN(C)C(C2CC3CCCCC23)=O)c(C)cc1Br c1(OC)cc(C)ccc1NC(C1CCC1CNC(C1(CO)COC1)=O)=O c1(OC)ccc(C(=O)N(CC(C)(C)NC(=O)CC(C)(C)C(F)F)C)cc1[N+](=O)[O-] O=C(CCCCCn1cnnn1)NC12CC1CN(C(c1nc(Br)c[nH]1)=O)C2 c1(C(N(CCCNC(=O)C=CBr)C2CC2)=O)ccc(C(F)F)cc1Cl N1(C(CC2CN(C(CNN(C)CCO)=O)C2)=O)CCC(N=[N+]=[N-])CC1.CCC1CC1 C(=O)(CCC1=NNC(=O)CC1)NCCOCCn1cc(C(CC)(C)OC)nn1 N1(C(C(c2cscn2)N(C)C)=O)CC2CC1(CNC(C1CC3(C1)CC3F)=O)C2 C1(NC2CN(C(=O)NC3(C(=O)OC)CC3)C(c3ncc[nH]3)C2)CCC2(CC2)CO1 N1(C(c2ccn(CCC)n2)=O)CCCC(CNC(=O)Cn2ccccc2=O)CC1 CC1COCCC1N(C)C(C1CCCN1C(=O)C(Cl)Cl)=O O=C(C1=CCCOCC1)N1CCC(c2cccc(C(F)(F)F)c2)C1 N1(C(CCC2CCC(C)O2)=O)CCC(C(=O)N(C)CC2(C)CC2)C1(C)C N1(CC(=O)Nc2nnc(O)s2)CCC(CNC(c2nccc(C(F)F)n2)=O)CC1 C(=O)(C(C(C)C)NC(=O)C(C)=C(C)CC)NC(CC#C)CO N1(CC(=O)NC2C(NC(COCCC(C)C)=O)C2)CCCCC1 C1(CC(=O)N(CCN(C(=O)COC2CCOC2)CC)CC)COCC1O C1(C(=O)NCCOCCC2CC2)CSCCN1C(C1CN2CCC1C2)=O Nc1cc(C(N2CCC2CNC(=O)C(F)C2CC2)=O)cc(C(F)(F)F)c1 c1(C(N(C2CN(C(Cc3nnc(C)o3)=O)C2)C)=O)c[nH]c(=N)c2[nH]ccc12 C1(C(=O)NCC2(C(C)(C)C)CCN(C(c3cc(F)c[nH]3)=O)C2)CCCCC12CC2 c1(CC(C)C)cc(C(=O)NCCC2CCN(C(C3CC3CF)=O)C2)ccc1F C(=O)(CCCCCn1cnnn1)N1C(CNC(c2c(C)snc2)=O)COCC1 c1(-n2cc(C(C(=O)OC)NCc3n[nH]cc3Cl)nn2)ccc(Cl)nc1 C(=O)(C(C)(C)C(=O)NCC1CN(C)CCN1C(=O)CCCCCNC(C)=O)NC C(C(=O)O)(C(C)OC)NC(Cc1cn(CC)nc1)=O c1(C(N2C(C3(O)CN(C(CCCOC(C)=O)=O)C3)CCC2)=O)cc(C)cc(C)c1 c1(C(N2CCC(C(C)NC(=O)C(C)(C)N(C)C)C2)=O)n[nH]c2c1CC1CC21 c1(C(=O)NC2C(NC(c3cc(Cl)sc3Cl)=O)CCC2)nccc2cccnc12 Cc1ccoc1C(=O)NCC(C)(C)CN(C(C)C(=O)NCC(F)(F)F)C N1(C(C2CC(CCNC(c3cc(CC)no3)=O)C2)=O)CCCC1(C)COC c1(C(=O)NC(C(CC)C)C(=O)NC)ccn2c(O)nnc2c1 C1(C(=O)NCc2nnc(C)s2)CN(C)CCN1C(=O)C(C)CC1CCCC1 c1(CC(=O)NCCCNC(C=CC(C)(C)SC)=O)nnc(-c2ccccc2)o1 C1(CNC(C(C)N(C)C)=O)CCN(c2ncc3c(n2)NC(=O)C3)CCC1(F)F C(=O)(CCC(=O)OC(C)(C)C)N(C)CC1(NC(C2CCCC2F)=O)CC1 c1(C(N2CC(N(C(c3cccc(CC)c3)=O)C)C2)=O)cc(N(C)C)cc(C#N)c1 Cc1cc(Cl)cc(N)c1C(=O)NC(C)C(C)NC(C1CC(N2CCCC2)C1)=O N1(C(c2c(C)ccc(C)c2)=O)CC2CCC(CNC(C3CC3F)=O)(C2)C1 C1(CN(C2CC(O)C2C)CC)CCN(C(=O)CC2CCCN(C)C2)CC1 N1(c2nnc(C)s2)CCC2(CCC2)C(NC(c2cc3c(o2)CCCC3)=O)C1 C1(C)(C(=O)NCC2CN(C(c3c(OC)csc3)=O)C(C)C2)CCCCNC1=O C1(CC)(NC(=O)CCn2cc([N+](=O)[O-])cn2)CCCN(C(=O)CCCC#CC)C1 N1(C(C2(CNC(C3=CCC(C)CC3)=O)CCC2)=O)CC2CCN(C)CC2C1 N1(CC(=O)N(C(C(=O)N(c2ccsc2)CC)C)C)CCC(C)C1 c1(C(N2C(CCNC(C3CC(C)(C)O3)=O)COCC2)=O)cc(O)cc(F)c1F N1(C(c2c[nH]nc2C2CCOCC2)=O)CCC(C2CCCN2C(=O)C2CC2)CC1 C1(CNC(=NCC2(OC)CCCCC2)NC2CC2)NC(=O)CC1(C)C C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2cc(F)c(F)cc2F)=O)CCC1(C)C C1(C(=O)NCCOCCCN(C)C(C2CC(=O)CCO2)=O)CC2(C1)CC2F c1(C(=O)NC2C3CN(C(C4C(COC)CC4)=O)C2C3)c(O)nnc2c1CCCC2 c1(C(=O)NCCC(=C)CNC(c2csnc2OC)=O)cnc2sccn2c1=O C1(CC(=O)NCC(CN(C(C=CC(=O)N(C)C)=O)C)O)CC2(CCC2)CO1 C(CCC(C)C)(C(=O)NCc1ccncc1F)NC(CC(C(=O)OC)C)=O n1(CC(=O)NCC(c2ccc(COC)cc2)O)cc2ccccc2n1 C1(C#N)(C(N2C(C3(O)CN(C(c4n(CC=C)ccc4)=O)C3)CCC2)=O)CC1(C)C C1(NC(C(=O)NCC)=O)CCC2CC1CN2C(=O)CN1CCN(C2CC2)C1=O C(=O)(CS(=O)(=O)C1CC1)N1C(C(=O)Nc2ccc(OCC)c(OC)c2)CC(F)C1 c1(N(S(C)(=O)=O)CC23CN(C2)C3=O)cnc([N+](=O)[O-])n1C.CC1CCC(=CC)C1 N1(C(COC(CC)(C)C)=O)CCC(C)C1CNC(=O)CSCCC#N N1(C(COC(C)C)=O)CC(CNC(=O)C(=Cc2c[nH]cn2)F)CC(C)(C)C1 N1(C(C2CC(C)(C)NC2)=O)CCCC2(CCCO2)CC1 C1(C(=O)NCC)(CC)CCCOC1.c12ccccc1C(C)C(=O)N2 C1(CC(=O)NCC(O)CNC(C2(Cl)CC2)=O)CC(CF)C1 C12(C(N3CC(C)(NC(c4cnc(C5OCCO5)s4)=O)C3)=O)CCC(F)(CC1)C2 N1(C(c2cnc(OCC)s2)=O)CCCOC(CNC(C2CCC(=O)C2)=O)C1 C(C(C)(C)CC(F)F)COC(C(C)N(C(=O)C(F)=CCCF)CCC)=O C(=O)(C1=CCCCC1C)NCC1(NC(c2cnc(SC)n2C)=O)CC1 C(C)(N=c1[nH]c(=NC(CC)C2CCC2)[nH]c2c1COCC2)c1c(C)cccc1Cl N1(C(C(C)NC(C)=O)=O)CC(CNC(c2ncccc2CO)=O)C(C(F)(F)F)C1 C(=O)(C1Cc2ccc(F)cc21)N1C(CNC(C2(SC)CC2)=O)CC2CC21 Cc1cnc(CCCNC(=O)CN(CC(C)C)C(c2nc(O)n[nH]2)=O)[nH]1 CCCCC(O)CNC(=O)CSCCNC(=O)CCc1cnc(C)o1 c1(NCC(=C)CC)cc(NC(c2cccnc2)CC2CCOC2)ncn1 C1(N(C(C(C)OCCOC)=O)C)CCN(C(c2cn(C)nn2)=O)C1 CC1CN(C(=O)C(C(C)O)N(C)C)CCC1NC(=O)CCC1CCCN1C N1(C(CN(C)S(N)(=O)=O)=O)CCC(O)C(NC(=O)CC2CC3CCC2CC3)C1 C1(CC(=O)NC2C(F)CCN(C(c3c(C)cccc3)=O)C2)CCC12CCOCC2 N1(C2CN(C(C34CC(C)(C3)C4)=O)C2)CC(Nc2c(NC(N)=O)cccc2)CC1=O C1(CC(=O)NCC(=O)NCC=C)CCCN(C(C23C=CC(CC2)C3)=O)C1 c1(C(=O)OC)cccc(CN2CC3(CC3)CC2C(=O)Nc2cccc(Br)n2)c1C c1(C(=O)NCC(CO)NC(c2c(C)nc(C)[nH]2)=O)cc(Cl)cc(C(F)(F)F)n1 CN1CCC2(CCCCN2C(CN=[N+]=[N-])C(=O)NC2CCOC2)C1 N1(C(c2csc(C)c2C)=O)CC2CCC(C1)N2C(c1nn(C)c(Cl)c1Cl)=O c1(CNC2C(NC(C)=O)CCCC2)nc(O)c2cnn(C)c2n1 N1(C(C2(CCCC)CC2)=O)CCN(CC(=O)Nc2cc(OC(C)C)ccn2)CC1 c1(CNC2C(C(=O)Nc3ncnc(OC)c3OC)C2)c[nH]c2ncc(Cl)cc12 C1(NC(C(C)NC(C2CCCCC2)=O)=O)(CO)CCCN(C(=O)Cc2cc[nH]n2)C1 N1(C(C2(C(C)C)COC2)=O)CCCN(C(C2CCC23CCOCC3)=O)C(C)C1 N12CCN(CC1)c1cc(ccn1)CNC(=O)C1CN(C(F)C2=O)C1.C(C)(=O)N.CO C12(C(N(C)CC3CCCN(C(c4csc(Cl)c4)=O)C3)=O)CCCC(C)(C1)OC2 c1(C(N2C(C(N3CCC(F)(C(N)=O)C3)=O)CC2)=O)c[nH]c2ccncc12 N12CCC(CC1)C2C(=O)NCCC1CC1.c1(SCCl)cnn(-c2ccccc2)c1 n1(C(C)C)cc(C(=O)NCCn2cc(C(=O)NCc3cn(C)cn3)nn2)nn1 c1(C(=O)NCCC2N(C(C(CC#C)O)=O)CCC2)cnc2onc(C)c2c1 C(C(O)C(=O)NCC1(NC(=O)COCc2ccnn2C)CC1)N(C)C N1(C(C(c2ccnn2C)NC2CCN(CC(=O)NC(C)C)C2)=O)CCC(C)(F)C1 C1(NC(=O)NC2(CC(C)C)CCOCC2)CCC(=O)N(c2ccccc2)C1 C1(NC(c2c(C)nc(C3CC3)o2)=O)CC2(CCN(C(C3CCCC3C)=O)C2)C1 N1(C(CC(C)n2ccnc2)=O)CCC2CC1CN(C(C1(CCF)CC1)=O)C2 C1(C(N(CC(=O)NOCC(O)CO)C(C)C)=O)CC(C)CC(C)C1 C1(C(=O)NC2COC3CCCCC23)CC2(CCCCCC2)N1 c1(C(=O)NC2CN(C(c3ccc(CC)cc3)=O)C(C)CC2)ncc(C#N)cc1C C1(CNC(C2C(C)(C)C(F)(F)C2)=O)CCCC2(CN(C(C3CCS3(=O)=O)=O)C2)O1 CCCCC(CN=c1cc(C)nc(Cl)[nH]1)NC(=O)C(C)OCC1CCC1 c1(CSCCCNc2c(Br)cnc(C(C)C)n2)cc2ccccc2o1 N1(C(C2(CC)COC2)=O)CCC2(C1)CN(C(c1ccc3cc[nH]c3c1)=O)CCO2 c1(NC(C2CCN(C(c3ccc(O)cn3)=O)CC2)=O)cccc(C(F)(F)F)n1 c1(OC)cc(NC2CC(CNC(C3(O)COC3)=O)C2)nc(C(C)C)n1 C1(C(C)C)CN(C(c2cccnc2)=O)CCC1NC(=O)C(C)(C)C1CC1 N1(C(C2N(C(c3c(C)n(C)cc3)=O)CCCC2)=O)CC2CC1CC2CF C1(C(N2CC(C3(NC(C=C(C)c4ccco4)=O)CC3)C2)=O)CCC2(C1)CC2(F)F Cc1ccc(Cl)c(F)c1NC(=O)NCC1CC(O)C1(C)C O=C1CC2(CCCN(c3nnnn3CCc3cncs3)C2)Oc2ccccc21 c1(C(N2CC(F)(CNC(C3(CC(C)C)CC3)=O)C2)=O)cn(C)c(=O)nc1O N1(C(CC2CCC(C)C2)=O)CC(C2(NC(c3cccc(C(C)(C)C)n3)=O)CC2)C1 C12(C(N3CC4C(OCC)C4C3)=O)CCCC(COC)(C1)OC2 CC1CC(C(N2CC=CC2(C)C(N2CCC(N3CCOCC3=O)C2)SC)=O)CN1C C(C(=O)NC(C)(C)C)(C1=CCCCCC1)N1CCN(C(COC)=O)CC1 N1(C(C2C(C(N)=O)C2)=O)CCCC1C=CC(=O)NCCn1cnccc1=O N1(C(c2cn(C)nc2O)=O)CCC(NC(=O)CC2CCCOC2)C(O)C1 n1(CC(=O)NC2(CO)CN(C(c3ccnn(C)c3=O)=O)C2)cnc2ccccc12 N1(C(C(CC)COC)=O)CC(C(N2CCCC2CC(=O)OC)=O)CC12CCC2 c1(C(=O)NC(C)CNC(=O)Cc2ccc(F)cc2F)ccc2c(c1N)CCCC2 C1(C(=O)NCC2(F)CN(C(c3cccc(CC#N)c3)=O)C2)CC2CCC1NC2=O CS(C)(=O)=Nc1ccc(C(N2CC3CC3(NC(=O)CC3CCCC3)C2)=O)s1 N1(C(C2CCN(C)CC2)=O)CCCCCC(NC(c2cnc(O)c(Cl)c2)=O)C1 CC1CCC(c2ccccc2)CN1C(=O)CCC(F)F.c12cn(nn1)C2C C(=O)(C#CC1CCOC1)NC1C(C)CN(C(C2CC(S(C)(=O)=O)C2)=O)C1 CCC(CC(F)F)C(=O)N1CCC(CCNC(=O)C(c2cccnc2F)(C)C)C1 c1(O)cccc(Cl)c1.c1(C(C)(F)F)cccc(F)c1.C12CC(C1)NC(=O)N2 N1(C(CC(C)C2CC2)=O)CC2CC1CN2C(C1CC1(C)C)=O Cc1cncc(C(N2CC=CC2CNC(=O)Cn2cc(C(F)(F)F)nn2)=O)c1C n1(C(C)C)cnc2c(NC3CCCC3CO)[nH]c(=NC(C)c3ccnn3C)nc12 C1(C(=O)NC(C)Cc2cn[nH]c2)CC(N=[N+]=[N-])CN1C(c1n[nH]c2c1CCC2)=O N1(C(c2c(C)nc(N)cn2)=O)CC2CCC(C1)C(NC(c1cccc(F)c1)=O)C2 CC1=C(C(=O)N2CCCC3(NC(c4n[nH]cc4Br)=O)CC3C2)C(=O)OC1(C)C C1(CC(=O)NCC(CN(C(C2CC(O)(CC#C)C2)=O)C)(C)C)CCCCC1C C(CCN(C)C)(C(=O)NCCCCN=[N+]=[N-])NC(C(n1c(C)ncc1)C)=O O=C(C1CCc2cc(F)ccc21)NC12CC1CN(C(=O)CCC1CC(F)(F)C1)C2 C1(NC(c2c(C(C)C)con2)=O)CC2CC1N(C(c1ccc(C(C)(C)C)s1)=O)C2 C1(C(=O)NCCCCCNC(C2CC(OCC)C2)=O)CCCC(C#N)C1 Cc1ccc2c(c1)C(NC(c1cnc(C)[nH]c1=O)=O)CCC2 c1(C(N2CC3CC3(CNCc3ccccn3)C2)=O)cc(I)ccc1O Cc1nc(Br)sc1C(=O)Oc1cccc(CN2CC3C(CNC(C)(C)C)C3C2)c1 c1(CNC(=O)NC(c2ccc(Cl)cc2)C(N)=O)cc2n(n1)CCCO2 CCC(CC)CCCC(=O)N(CCCCCNC(=O)C(C)c1ncco1)C CC(C)CC(O)C(=O)NC(c1cccnc1)CNC(C1(C)CC1C)=O c1(NC(c2ccc(C)s2)CC)cc(NCCN2CCC(F)C2)nc(COC)n1 N1(C(c2c(CNC(C3(C)CN(C)C(=O)C3)=O)nnn2C)=O)CCn2nccc2C1 C1(C(N)=O)(NC)CCN(c2ncnc(NC(C)CC(C)O)c2C)CC1 c1(-c2n(CCC#C)c(N3CCC(COC)C3)nn2)nc(C2CC2)n2ccccc12 c1(NC(C2N(S(CCC)(=O)=O)CCC2)=O)cccc(NC(=O)CC(C)COCC)c1 N1(C(C(CNC(C(CC#C)C2CC2)=O)CC=C)=O)CCC(C)OC(C)C1 C1(C(=O)NCC2(O)CN(C(CC(C)(C)C)=O)C2)CCc2c[nH]nc2C1 CCC(CC(=O)N(C(C)(C)C#N)C)C1CC1.C12(CC1)CC(=O)N2 N1(C(CCC(=O)c2ccccc2)=O)CC(F)(F)CC1CNC(=O)CC1CC12CC2 C1(N2CCN(C)CC2)(CN(C(c2nccs2)C)C(C)=O)CCCCC1 c1(CNC(Cc2cc(C)no2)=O)ncccc1C(=O)NCC1C=CCC1 N1(C(C2CC=C(C)CC2)=O)C2CC1CN(C(=O)Cc1cn3ccsc3n1)C2 C#Cc1ccc(C(N2CCC(C)(CNC(=O)Cc3cnns3)CC2)=O)c(F)c1Cl c1(CC)ccc(NC(=O)C(c2cccs2)NC(=O)CSCC(=O)OC)cc1 C(C(C)CCCC(C)C)N(C(C)C(=O)NOCCO)C(CC(C)C)=O c1(N(C)Cc2n[nH]c3ccccc23)nc(=N)[nH]c2ccccc12 C1(CNC(C2(CCC)CC2)=O)(NC(=O)CNC(=O)C(C)(C)C)CCCCC1C CC(CNC(C1SCCS1)=O)CC(=O)NC(CO)(CO)CO c1(C(N(C(C(N2CCC(CC=C)C2)=O)CC)CC)=O)cnc(C)cn1 CC1CN(C(=O)CC2CCC(O)C2)CCN(C(c2c[nH]c(C#N)c2)=O)C1 N1(C(c2nccc(OC)c2F)=O)CC(C)OC2(CCN(CC#N)C2)C1 O=C(CC(C(F)F)NC(c1cnn2c1CCC2)=O)Nn1nnc2c1CCCC2 c1(CCC(=O)NC(CC)CN(C(=O)Cn2nnc(=O)[nH]2)C)cn(C)nc1C c1(CC)cc(C(=O)N(C(C)CNC(=O)Cc2ccccc2O)C)cc2c[nH]nc12 c1(SCC)ccc(C(=O)NCC(C)NC(=O)COc2cc(C)ccc2F)c(Cl)c1 C(=O)(CC(C)P(C)(C)=O)NCC(C)(CNC(c1coc(C)c1)=O)OC CCCCCCn1nnnc1C(C1(C)CCCO1)(C)NCC(C)(C)C1CCCC1 c1(C(=O)NC2CC(CNC(c3cc(C)c(Cl)s3)=O)C2)cc(C2CC2)ccc1F CCCCCCCC(=O)NCC(O)CNC(c1ccc(Cl)nc1O)=O C(C(C)(C(=O)N1CC(O)(CNC(=O)CCC(=O)c2ccc[nH]2)C1)OC)OC C1(C(=O)NCCCN2CCCC2=O)(NC(C2CC(C)C2)=O)CCCC1C c1(-n2cc(CC3CCN(CC4=CCCC4)C3)nn2)c[nH]ccc1=O C(=O)(CC(C)(C)C#N)N1CCC(N(C(=O)C(C)Cc2ccco2)CC(C)C)CC1 c1(CC(=O)N(CC(C)NC(C2(C=C)CC2)=O)CC)ccc(Br)c(Cl)c1 c1(C(N(CC(CN(C(=O)CCC2OCCO2)C)O)C)=O)cnc(S)[nH]1 CCCCCC(O)CNC(=O)CCC(C)NC(C1CCC1C(=O)OC)=O C1(C(=O)NC(C2(O)CN(C(C3CCC4(CC3)CC4)=O)C2)C)CCC2CC2CC1 c1(C(=O)NCC2N(C(CC(C(C)C)C)=O)CC2)cc2cc([N+](=O)[O-])ccc2[nH]1 c1(C(=O)NC(C=C)C2CCC2)ccc(CN=c2nco[nH]2)cc1 C1(S(C)(=O)=O)(NC2CC(C)(OC)C2(C)C)CC(F)(F)C1.c12cc(sn1)C(=O)O2 C1(C)(C(=O)NCCC(C)O)CN(C(c2cncc(Cl)c2)=O)C(C)(C)C1 N1(C(c2ccsc2Cl)=O)CCSCC1c1ccccc1 C12(CNC(C(C)(C)OCC)=O)CCC(CC1)CN2C(=O)CCc1ncccc1C C1(N(C(C2C(OC)CC2)=O)C)CCC2(CC1)CCN(C(c1ccnc(O)c1)=O)C2 C1(CNC(c2c(C(C)NC(=O)C3CC3)noc2)=O)COCC1O C1(CNC(C(CC)SC)=O)CN(C(=O)C(O)C(=O)OC(C)(C)C)CCC12CCC2 N1(C(C2N(C(C(COC)O)=O)CC=C2)=O)CC(OC(C)=O)CC(C)C1 c1(C(=O)NC2C(C)CN(C(=O)CCC3CCCO3)CC2)ccc(N)c(Cl)c1O C1(C(N2C(CC(=O)N(C)C)CCCC2)=O)CCN(C(=O)C(C)(C)C)CC1O C1(NC(C(SC)SC)=O)CN(C(=O)C=CC(=O)N(C)Cc2ccccc2)CCO1 C1(NC(C(CN(C)C)O)=O)CC=C(C(=O)NC(CCO)C2CC2)C1 N1(C(CCSCCC)=O)CC(CC(N2CCCCC2C2CC2)=O)C2(CC2)C1 c1(CNC(=NC)NCC(=C2CCOCC2)F)ccc(F)c(C)c1 N1(C(CN(C)C2CC2)=O)CCC(NC(c2coc(Cl)c2)=O)C12CCC2 CC1(C)CCCC(O)(C(N2CC3(CCC3)CC2CNC(=O)CCCCO)=O)C1 c1(CNC(C(C)SCC)=O)cc2c(cn1)COCC2.C12CCC13CN(C3)C2=O N1(C(c2cnc(C)o2)=O)CCCCC(C(=O)NCc2ccc(Cl)o2)C1 C1(CNC(C(CC)(C)CC)=O)CCC2(CN(C(=O)C(C)Nc3nc(C)cs3)C2)O1 c1(C(C2CC(NC3C=CS(=O)(=O)C3)C2)O)ccccc1Cl c1(NCCC=C)nc(N2CCc3c([nH]c4ccc(Br)cc34)C2)nc2c1cnn2C C#Cc1ccc(Cl)c(C(=O)NC2CN(C(C3CCOCC3(C)C)=O)C2)c1 c1(OC)ccnc(CN(C(=O)C(=O)NC2CCC(=O)N2)Cc2ccc(F)cc2)c1 C(CO)(CCCCNC(c1cnc(O)c(OC)c1)=O)NC(c1cc(OC)ns1)=O c1(C(=O)NC2CN(C(CCCSC)=O)CC2(C)C)cc(C)c(O)c(N)c1 Cc1c(Cl)ccnc1C(=O)NCC1CC(C)N(C(c2coc3c2COC3)=O)C1 C1(C(=O)NCC(O)C(=O)NC2CCN2C(C)(C)C)(CC)CCCCC1 c1(C(=O)NC2CN(C(CSCCC(C)C)=O)C(C)C2)cc(C#N)n(C)n1 C(=O)(N=c1cc(C)n(CCNC)[nH]1)C1N(C(c2ccc(C)cc2C)=O)CC(C)(C)C1 c1(C(=O)NC(C(=O)NC(c2cnc[nH]2)C)c2ccoc2)cccnc1 c1(C(N(CC(=O)O)CCC)=O)ccccc1-n1cc(-c2cncc(Cl)c2)nn1 N1(C(C2(C)C(C(=O)OC)C2)=O)CCCOC(CNC(C2CC(C)(F)C2)=O)C1 C1(C(N2CC(F)(CNC(c3cc(OC)no3)=O)C2)=O)CCC(C)(C)OC1 n1(NC(N2C(C(N3CC4N(C)C(CC4)C3)=O)CCC2)=O)c(=O)oc2ccccc12 N1(C(C2(COC)COC2)=O)CCC(C2CCN(C(C3(COC)CC3)=O)CC2)CC1 c1(C(C)C)cccc(N2CC3C(CNC(=O)CC4CCCC4C)C3C2)n1 C1(C)(C(N2CCC(C(N(C)CCOC3CC3)=O)CC2)=O)CCCCC1(F)F c1(CNC(c2n(C)cc(Nc3cc(F)cc(C#N)c3)n2)=O)cc(Cl)c(Cl)cc1O c1(OC)cccc(C2CCN(C(=O)CNCc3cc(-c4ccoc4)on3)C2)c1 C(=O)(CC(C(F)(F)F)NC(c1cccn2cncc12)=O)N1C(C(C)O)COCC1 c1(C(C)C(=O)NC(C(=O)NCCN=[N+]=[N-])C2(O)CCC2)ccccn1 C12(NC(CCC=CC)=O)CCC(C(=O)NCC(C(C)C(C)C)N(C)C)(CC1)CC2 c1(CC(N2CCCN(c3ncc(Br)c(O)n3)CC2)=O)ccc(Br)cc1Cl CCCCCCC(O)CCC(=O)N1CCCC1CNc1ncnc2cnn(C)c12 NS(=O)(=O)CC(=O)NC1CCC(NC(=O)COc2cccc(-n3ccnc3)c2)C1 C=CCC(CNC(=O)Cc1csc(Cl)c1)NC(C1(O)CC1)=O Cc1cccc(CN2CCC(C(N3CC4CCC(C3)O4)=O)C2)c1Br N1(C(=O)OCC)CCCC(CC(=O)NCC2(n3ccnn3)CC2)CC1 N1(C(C(C)OC)=O)CCCN(C(c2ccc3sncc3c2)=O)CC1CO c1(C(N2C(CNC(C3C(=C)CC3)=O)CN(C)CC2)=O)ccc(CC)c(CC)c1 CN=c1[nH]c(C(=O)OCc2nccc(C(F)(F)F)n2)cs1 C1(C(=O)NC2(C(=O)NCCCC(C)(C)OC)CC(F)(F)C2)CC2CC1CC2O C1(C(=O)NC2CCN(C(COC(C)=O)=O)C2C)CCCC2(CC2)C1 C1(CC(=O)N(C)CC2CCN(C(=O)CNC(c3cscn3)=O)C2)CCC12CCC2 C1(NC(c2nc(C)sc2C)=O)CCC2(CC1)CN(C(=O)Cc1ccc(N)cc1)C2 N1(C(c2nc(Br)cs2)C(=O)NCc2cccs2)CCC(N2CCOCC2)C1 C1(NC(C(CCCC)F)=O)CN(C(c2cn(C)nc2O)=O)CC2(CCC2)C1 S(=O)(=O)(c1cccc(=NCC2CC2Cl)[nH]1)NCCCN1C(C)(C)COCC1 c1(NCCN(c2ccccn2)C)nccc(=NCC2CCCSCC2)[nH]1 Cc1nc2ccc(C(=O)NC(CO)CCCNC(=O)C3=CS(=O)CCC3)cc2[nH]1 N1(C(CC2N(C(CC(C(C)=O)(C)C)=O)CCC2)=O)CCc2nncn2CC1 C(=O)(C(CCSC)NC(=O)CCOC(C)=O)NCC1(CCC)CCC1 Cc1cc(C)c(C(=O)NC2CC(CNC(c3sc(Cl)c(Cl)c3C)=O)C2)c(C)c1 N1(C(c2c(CC)csc2)=O)CCC(O)(CCNC(=O)CC2CCCOCC2)C1 N1(C(=O)CCC2CCC(=O)N2)CC2CCC(C1)N2C(=O)CC1CC=CCC1 N1(C(C(C2CCCC2)OC)=O)CC(C(=O)NCc2ncccc2O)CC(C)(C)C1 N1(C(C(C(C)C)NC(C)=O)=O)CCN(C(c2ccoc2)=O)CC12CCC2 N1(C(CCC=CCC=C)=O)CCC(NC(C2CC(C3CC3)=NO2)=O)C2(CCC2)C1 CCC(CCC(=O)NCC(F)C(C)(C)O)NC(c1n[nH]cc1C1CC1)=O C(CC(F)(F)C(F)F)n1cc(COC(C)C(=O)NC2(c3ccccc3)CC2)nn1 C1(CNC(c2sccc2F)=O)CCCC(NC(c2ccc(F)s2)=O)C1 C(=O)(C#CC(C)(C)CNC(C1CCCC(=O)C1)=O)N(C)Cc1cc(C)on1 C1(NC(C2C(CNC(C(COC)C)=O)C2(C)C)=O)CCC2(CC)CC1CC2 N1(C(c2cnc(C)o2)=O)CC(NC(=O)C=Cc2nccs2)C(C)(C)C1 N1(C(CCC(C)OC)=O)CCCOC(CNC(c2cc(F)c[nH]2)=O)C1 c1(C(=O)NC2(CNC(C3C(CC)C3)=O)CCOC2)cccn2cc(C)nc12 C=C1CC(c2ccccc2)(C(=O)N(C)CC2CCCN2C(=O)C(F)CC2CC2)C1 N12CC(CC(C)C1)NC2=O.C1(CN(C(C)(C)C)CC=C)CC(C)C1 N1(C(CCC(=O)NC)=O)CCC(NC(c2cc(C)nn2C2CCC2)=O)C(CO)C1 N1(C(C=CC=CCCCCC)=O)CCC(N(C(C2COCCN2C)=O)CC)CC1 N1(C(c2cc(SC)oc2)=O)CCN(CC(=O)NCc2csc(O)n2)CC1 c1(C(N2CCN(C(C3(C#C)CC3)=O)CC2C)=O)cc(F)cc2nccnc12 C1(NC(C(CC2CC2)NC(C2(C3CCCO3)CC2)=O)=O)CCCN(O)C1=O N1(C(CCOCCOCC)=O)CC(C(=O)NCC(C2(O)CCC2)C)C(C(C)C)C1 c1(NC(C(C(=O)OC)(C)C)C)ncc(-c2cccc(C(F)(F)F)c2)cc1C#N N1(C(c2nnc(C)s2)=O)CCSCC1CCNC(C1COCCO1)=O N(C1CCc2c(C)ccc(Br)c21)S(c1c(Cl)ccc(C)c1)(=O)=O C(N=c1[nH]c(=NCC2(C)CCC(=O)N2)[nH]c2cccnc12)C1(CO)C(C)(C)C1 CC(C)C(F)(CNC(=O)Cn1ccnn1)C(=O)NCC1COCCN1C CC#CCC(C(=O)N1CCS(=O)C(C)C1)NC(=O)C(C(C)(C)C)OC C12(NC(c3cccc(OC)c3OC(C)C)=O)CCCN(C(=O)CC#N)CC1C2 N1(CCNC(CN(CC)CC)=O)CCCN(C(c2cnncc2NC)=O)CC1 C1(C(=O)NCCN(C(CC)C)C)C(C)CCN1C(=O)C=Cc1cc[nH]n1 C12(C(=O)NCc3cnn(C)c3C(N3CCOC4(CC4)C3)=O)CCCC1C2(F)F c1(C(=O)NCC(CO)NC(C(C2CC(F)(F)C2)OC)=O)sccc1C(C)(C)C c1(CC)onc(C)c1C(N1CC(NC(=O)CCCCOC)C(C)C1)=O N1(C(c2c(C)cns2)=O)CCN(C(c2csc(-c3cn[nH]c3)n2)=O)C(C)C1C C1(CNC(C(CCC)C)=O)C2CCC(C2)N1C(c1ccnn1C(C)C)=O CC#CCC(C(=O)N1CCCNC(=O)C1)NC(=O)C(C)CCOC c1(OCC)ccc(C)cc1C(N1CC(n2cc(C(C3CC3)OC)nn2)C(C)C1)=O N1(C(CN(CCOC)C)=O)CCC(CO)C(NC(c2cccc(Cl)c2Cl)=O)C1 CN1CCN(C(C2CCC(O)CN2C)=O)C(CNC(=O)CC(C)(C)C2CC2)C1 c1(C(N(C2CCN(C(CCOC)=O)C2)C)=O)cc(S(N)(=O)=O)ccc1O Cc1c(Cl)sc(Cl)c1C(N1CCC(O)(CNC(c2cnc3n2CCC3)=O)C1)=O CCC(C)(C)CC(=O)N1CCC(CNC(=O)CC2CCOC(C)(C)C2)(OC)C1 Cc1cc(C(=O)NC2C=CC(CC(=O)N(C3CCCCCC3O)C)C2)cnc1O C(CCCCCNC(=O)CCCCN(C)C(C1C2CC(=O)CC12)=O)N(C)C c1(C(=O)NC2CC(NC(=O)C3=CS(=O)CCC3)C2)cncc2ccccc12 C1(C(N(C(C)CNC(c2ccncc2C)=O)CC)=O)CC(=O)c2ccccc2O1 c1(OCCSCC)ccccc1Cl.CCC1C(=O)O1 c1(C(N2CCOCCC2C(F)F)C(=O)NCCSC)cc(F)cc2cccnc12 C(=O)(CC(CCC)NC(C1(CO)CCCC1)=O)N(CC(C(=O)OC)C)C C1(C(=O)NC2CN3CCCC2C3)C2CCCC2CN1C(c1cccc(F)c1)=O c1(SCC)cnccc1C(=O)NCC(CNC(=O)CC1CCC(=O)N1C)OC c1(NC(CC(C)O)=O)cccc(NC(C2(C(F)F)CC2)=O)c1 N1(C(C2C(COC)C2)=O)CC2CCC(NC(c3cnnc(Cl)c3)=O)CC2C1 N1(C(c2[nH]cc(C)c2C)=O)CCC(NC(C2CCCC(CF)C2)=O)C12CC2 Cc1nc(N2CCC(C(=O)NC(Cc3ccccc3)CO)CC2)ccc1F c1(C(N2CC(C)N(C(=O)CCC3CCCCC3)CC2)=O)cnc2[nH]ccnc1-2 CC(C(C)(C)NC(=O)CC1CCC1(C)C)NC(=O)COc1ccccc1 c1(OC)cc(C(N2CC3C(C2)N3C(c2nc(Br)cs2)=O)=O)ccc1OC(C)=O n1(Cc2cc(C)on2)nnc(C(=O)NC2(CCCNC(=O)CNC=O)CC2)c1C C(=O)(C(C)CC(=O)NCC1CCN(C(C2CC(C)CCO2)=O)C(C)C1)OC c1(CC)cc(O)ccc1NC(=O)CCN(C(=O)C(F)n1ccnc1)CC c1(OC)ccc(OC)c(C=CC(=O)NCC2CCC2NC(=O)C(C)NC(N)=O)c1 c1(OCC(N2CCCC2Cn2cc(C3(CO)CCC3)nn2)=O)ccc(Cl)c(F)c1 N1(C(CCn2ccc(C)n2)=O)CCC(NC(=O)CCc2ccc(C)s2)CC1C C1(C(=O)NC2CC(OC)CN(C(C3CC(=C4CC4)C3)=O)C2)(CC)CCC(O)CC1 C1(C(=O)NC2C(CNC(c3nc(C)n(C)n3)=O)CC2)C2CCC1(C)C2(C)C N1(C(c2ncn(C(C)C)c2)=O)CC(CNC(=O)CNC(=O)C(C)(C)C)C(C)(C)C1 C1(CNC(C2C(=C)CC2)=O)CN(C(c2ccc(C(C)(C)C)nc2)=O)CC1C CCC(C)CCCCC(=O)N1CCC(C(=O)NCCCC(O)CO)(OC)C1 Cc1ccc(O)c(C(=O)NC2CC3CC2CC3C(=O)NC(C)CC(N)=O)n1 c1(CC)nc(=NCCC2CCCN(C(=O)CC(c3ccc(OC)cc3)C)C2)s[nH]1 Cc1ccnc(C(=O)NCC(CNC(c2ccccc2C(F)(F)F)=O)CO)n1 C1(CN(C(c2cc(C)on2)=O)C)CCCC(NC(=O)COCCC(C)C)C1 c1(NC(C2CCCC(O)C2)c2n(CC(=C)C)nnn2)cc(C(F)F)cc(CC)c1 C=C=CCCC(=O)NC1CN(C(C2CCC(=O)N2CC(F)(F)F)=O)CC1OC c1(CC(=O)NCCC2(CNC(c3sccc3C(F)F)=O)CC2)cccc(Cl)c1F C(=O)(N=c1cc(C2CCC2)nc(O)[nH]1)C1CC2(CC(N(C)C3CC3)C2)C1 C1(OC2CC2)CCN(C(=NCCNC(=O)OC(C)(C)C)NCC2=CCCOC2)C1 c1(CC)onc(C(=O)NCC)c1C.C1(=O)C(CC2CCCC2)OC(=O)CC2CN1C2 Cc1nc(C2CCC2)sc1C(=O)NC1(C)CN(C(C2CC23CCC3)=O)C1 C1(NC(CCOCC)=O)CCCC2CN(C(c3ccccc3CN(C)C)=O)CC12 Cc1sc(C(=O)N(CC(C)NC(C2CC(C)(C)O2)=O)C)nc1-c1ccc(Cl)cc1 c1(NCC23CC(NC(=O)C=C(C)C)(CO2)C3)ccc(C(=O)OC)c(C(C)=O)c1 CC1CN(C(c2ccc(C3CC3)s2)=O)CCC1CNC(=O)CCF c1(OCC)ccc(Cl)c(C(=O)N(CCNC(=O)CSc2cccs2)C2CC2)n1 C1(CN(C(=O)C(C)NS(C)(=O)=O)C)CCCN(C(=O)C(C)(C)F)C1 c1(CC)ccc(C(=O)NCC(F)CNC(=O)C(CC)SC)c(F)c1 C1(C(=O)NC(CNC(CC(=O)OCC)=O)CC)CCCC(C(N)=O)CC1 C1(NC(C(C=C)O)=O)CC2CCC1(C(N1CC(S(N)(=O)=O)C1)=O)C2 c1(C(=O)OC)c(C)oc(C)c1C.N1(C(C)=O)CCOC(CC)C1 CCC(CCOC)C(=O)NCC1CN(C(c2sc(F)cc2C)=O)CC1C c1(C(N(CCOCCNC(CC(CCC)O)=O)C)=O)cnn2c1OCCCC2 S(=O)(=O)(c1cccc(C(=O)O)c1)NC(c1c(OC(C)C)cc(Br)cn1)=O c1(OC)ncc(NC(C2(CNC(C3C=CCCC3)=O)CCC2)=O)cn1 c1(C(=O)NC(CC)CNC(c2cnn3c2CCC3)=O)cnc(OC)cc1C(F)F C1(CNC(C(C)C#N)=O)CC2CCC1N(C(C1(C)CCCS1(=O)=O)=O)C2 CC(C)CC(C(=O)N1CCC1CN=[N+]=[N-])NC(=O)C=CC(=O)N(C)C O=Cc1sc(CN2CC3(CCN3C(c3cc(F)ccc3I)=O)C2)c(Br)c1Br c1(C(=O)NC2C(Cc3nc(CNC(c4c(OC)n[nH]c4)=O)sc3)C2)sc(F)cc1C c1(C(N2CC(NC(C)=O)C(C#N)C2)=O)cc(F)ccc1[N+](=O)[O-] c1(N(C)Cc2ccc(C)c(Cl)c2)nccc(=NCC2CC(C)(C)CCC2O)[nH]1 C(CC(C)C)(C(=O)OC(C)(C)C)NC(CCC)(C)c1nnnn1CC1CCCO1 c1(OC)ccc(C(N2CCC(C(=O)N(C)CC3CC4C=CC3C4)C2)=O)cc1 C1(NC(c2ccc(CNC(C)=O)s2)=O)CC(O)CN(C(=O)C#CC2CCC2)C1 Cc1nn(CC(N2CCC(CCNC(C3CCCC3C)=O)CC2)=O)cc1[N+](=O)[O-] C(=O)(C(C)(C)C)N(C(C)CN(C(=O)CN(C(=O)C=C1CCC1)C)C)C.C(COC)N C1(CCNC(C(F)=CC)=O)CCCN(C(=O)CCOc2ccc(C(N)=O)cc2)C1 C1(CNC(C2C(=C)C2)=O)CC2(CCN(C(c3sc(Cl)cc3Cl)=O)CC2)CO1 C1(C(=O)NCCC(=C)CNC(c2cccc(OCC)c2)=O)CCCCC1C CCCC(C(N)=O)NC(C1C=CCN(C(=O)C=Cc2cc[nH]n2)C1)=O N1(C(C)C)CCC(CC(=O)NCCCOCCOCC2CC2)CC1.OC N1(C(C=Cc2cc(OC)ns2)=O)CCC(O)(CNC(=O)CC2CCC(O)C2)CC1 c1(OC)cc(C#N)ccc1C(N1CCCC1CNC(c1cccc(C)c1C)=O)=O c1(C(=O)NC(CC=C)CNC(=O)CC2CCCC2)cc(C)c(C)nn1 c1(C(N(C(CNC(COc2cncc(C)n2)=O)C)C)=O)nn(C)c2c1CSCC2 N1(C(C(C)OCC=C)=O)CC=CC(C(=O)NCC(COC)C(C)C)C1 C1(CNC(CC2CC(C)C2)=O)CCCN(C(C2(C#N)CC2C(F)(F)F)=O)C1 c1(NC(=O)NC23CC(C(=O)Oc4ccc(SC)cc4)(C2)C3)cc(CO)ccc1Cl C(=O)(CC(C(F)F)C(C)(C)C)NCC1CCN(C(C(CC(C)C)OC)=O)CC1 O=C1NC(=O)c2c(C(=O)NC3CCCN(C(=O)C(O)CN4CCCC4)C3)cccc21 CC1CCCC=C1C(=O)NC(CNC(=O)CN=S(C)(C)=O)CO CC(C)C(C)C(CNC(c1ccccc1Cl)=O)NC(C1CC(C)(O)C1)=O c1(CC)ncccc1C(=O)NCC1CN(C(=O)Cn2cncn2)CC1N(C)C c1(CNCC(c2ncc[nH]2)C)ccc(OCc2ccccc2)cc1F C1(C(=O)NC2C(C)CN(C(=O)CCC3CCCCC3)C2)Cc2nncn2C1 C(=O)(C(C)(C)CC(C)C)NC(C1OCCN(C(Cn2nc(C)oc2=O)=O)C1)C c1(-c2cn(CC(=O)NC3C(C(=O)O)C3)nn2)ccc(OCCO)cc1 c1(OCC)cccc(Cl)c1CC(=O)NC1CCN(c2cccc(Br)c2)C1=O CCC(C)CCC(O)CC(=O)NCC1CC2(CC2)CN1C(c1csc(C)c1N)=O C1(C(=O)NCc2cc(C(=O)NC(C)C(C)(C)C)no2)CC2(CCC2=O)C1 c1(C(=O)NCCC2(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2)ncnc2sccc12 Cc1n[nH]c(C)c1C(N1CCOC(CNC(=O)Cc2ccco2)C1)=O N1(C(C=C(COC)C)=O)CCN(C(=O)C(F)(F)CCN(C)C)CC1n1cccn1 CCCCCCCOC.c12nccc(n1)C(=O)NCCCN2CC Cc1ccc(C(=O)NC2CC(C)N(C(C3CCC=CO3)=O)C2)c(O)c1C c1(C(=O)NC2C3CN(C(c4cc(CC)n(C)n4)=O)CC32)cc2oc(C)c(C)c2[nH]1 c1(C(N(CC(C)CNC(=O)COC2(C)CCC2)C)=O)cc(S(C)(=O)=O)co1 C1(NC(C(C2CCOCC2)OC)=O)CCN(C(=O)C2=COCCO2)CCC1(F)F N1(C(CC2CCC(=O)O2)=O)CC(NC(c2nncn2C2CC2)=O)C2CCCCC12 C(=O)(C1CCCn2nccc21)NCC1(C)CCN(c2nnc(C3CCCC3)s2)C1 C(=O)(C1=CCN(C(c2cc(Cl)cn2C)=O)CC1)NCC(COC)O c1(SCCCN(CCCNC(c2ccnc(CO)c2)=O)C)ccc(F)c(F)c1 CC(O)C(F)(F)C(=O)N1CCN(C)C(C(=O)NC2CC(O)(CO)C2)C1 C(C(=O)N=c1ccn(C2CCC2)[nH]1)=C(C)CNc1c[n+]([O-])c(C)cn1 c1(CC(=O)NC2C(CNC(=O)CCOCC3CC3)CCC2)cc2c(s1)CCC2 N1(C(Cc2cc(OC)c(Cl)cc2)=O)CC2CN(C(C3C(C)C3C)=O)CC2(C)C1 C1(CC(=O)NCC2CCN(C(=O)Cc3cccc(F)c3O)C2)CCCCC1(F)F C(C1(C)CCOCC1)=CC(=O)NC1CCCN(C(c2nc(C)n(C)n2)=O)C1 c1(C(C(=O)NC2CC(C)(NC(Cc3nc(C)sc3C)=O)C2)C)c(C)nn(C)c1C CC1(C2CC2)CCCN1C(C=CC(=O)N(C(=O)CN1CSCC1=O)CCO)=O c1(C(=O)NC(CC)CNC(=O)Cc2cn(C)nc2C)cc(Br)ccc1C C1(N(C)C)CCc2ccccc2C1NC(C1CCCN(C(=O)C2CC2)C1)=O C(CC(C(=O)N(C)CCOC1CCN(C(c2oc(C)nc2C)=O)C1)OC)OC c1(C(N2CCC(CCNC(C3(COC)CCCC3)=O)CC2)=O)cccc(Cl)c1F C#Cc1cncc(C(N2CCC(C)(NC(c3cc(Cl)no3)=O)C2)=O)c1 CN1CC(C(=O)NC(C(=O)NC(C(N)=O)C2CCCC2)C2CCC2)CC1=O CCC1=C(C(=O)NC2CCCCC2NC(=O)C=Cc2scnc2C)SCCO1 c1(C(N)=O)cc(C(=O)NC2(CC(=O)NCC3(O)CC(CO)C3)CC2)co1 C1(NC(CC(CC)OC)=O)CCOC12CCN(C(c1cc(C)cnc1C)=O)CC2 C1(C2CC2)(NC(C2C(NC(C3CCCN(CC)C3)=O)CC=CC2)=O)CCCCC1 C1(C(=O)NC2C(C(=O)NCc3cc(CC)[nH]n3)CCC2)CCOC(C)(C)C1 c1(C(=O)NCc2c(CNC(C(COC)C)=O)cccc2)cnc2n1CC(C)CC2 S(=O)(=O)(C1(c2cn(CCC3CC(NC(=O)O)C3)nn2)CC1)NC c1(CC(=O)NCCCNC(C(c2ccc(F)c(F)c2)C)=O)c[nH]c2ccccc12 C(N=c1nc(N2CCC(C(N)=O)CC2)c2sccc2[nH]1)C1(N(C)C)CCCC1 c1(C(N2CCC(C)(CCOC)CC2)=O)cccc2c1CCC2=O CC1CN(C(=O)C(F)(F)c2cnnn2C)CC(C)CN1C(C1C2CCCC12)=O Cn1c(O)ncc(C(=O)NCCC2CN(C(C3CSCCS3)=O)C2)c1=O C1(F)(CNC(C2(CC=C)CCC2)=O)CCN(C(C2(CC3CCC3)CC2)=O)C1 c1(CNC(=O)COc2ccc(OCc3ccccc3)cc2)ccc(B(O)O)cc1 c1(C(N2C3C(NC(C4=C(C)CCCC4)=O)C(C3)C2)=O)ccc(C)c2cccnc12 N1(C(C(CCC)OC)=O)CC(C2CN(C(c3c(OC)ccc(Cl)c3F)=O)C2)C1 C1(CC(=O)OCC)CCCN(C(=O)Nc2sccc2OC(C)(C)C)CC1 Cc1c(Br)c(C(=O)NCC2(CCNC(=O)CNC(=O)C3CC3)CC2)nn1C c1(N2CCC(NC(=O)Nc3cccc(-c4nnco4)c3)C2)ccc([N+](=O)[O-])cc1 C(=O)(CC(C)c1cccnc1)NCC1CC(NC(C2(NC(C)=O)CC2)=O)C1 C1(NC(CC2CCN(C(C)C)CC2)=O)(CO)CCCN(C(=O)CC(C)F)C1 C(=O)(C1=CCOCC1)NCCSCCNC(CCOC)=O Cc1cccc2cc(C(N3CCN(C(=O)C(C)c4cnco4)CC3CF)=O)oc12 C1(CNC(c2cc(CNC(C(C)(C3CC3)OC)=O)no2)=O)CC(C)(C)CCO1 C1(CCC=COC(C(=O)NC)C)(CNC(CN(C)CC)=O)CCCC1 C(=O)(C(F)C(C)CNC(=O)CC(C)F)NCCCOCCCC C(c1ccco1)=C(C)C(=O)NCCCCC1CN(C(C2(C)CC2Br)=O)C1 c1(C(N2CCCC2c2ccco2)C(=O)NC)cncc(Br)c1 C1(C(N(CCN(C(C(C2CC2)SC)=O)C)C)=O)CCCCC1C(C)(C)C Cc1csc2c(C(N3CCCC(CN4CCOC(CN)C4)C3)=O)ncnc12 Cc1cnc(N2CCC(O)(C(=O)Nc3cc(F)nc(F)c3)C2)nc1Br CC(C)C(O)C(=O)NC12COC(CNC(C3CCCCS3)=O)(C1)C2 C(=O)(CC(CC)C1CC1)NCC(CC=C)NC(c1cncc(N(C)C2CC2)c1)=O Cc1nccnc1NC(C1CC1NC(=O)OCc1cn(CC(C)C)nn1)=O C1(C(=O)NCC(CCC=C)(C)C)C(C2CC2)CCN1C(=O)CCC(C)=O Cn1nc([N+](=O)[O-])cc1C(N1CC2C(NC(C3(CC(F)F)CCC3)=O)C2C1)=O N1(C(CCC2C(C)=NOC2=O)=O)CC2(CCCC2NC(=O)CCC(C)O)C1 C(=O)(C1=C(Cl)CCCC1)NC1C(NC(Cc2ccc(OC)c(F)c2)=O)C1 C#C[Si](C)(CCC)c1ccccc1N(C(=O)CC(c1ccccc1)N(C)C)C O(NC(=O)C(C)(F)F)CC(=O)N(C(C)C)Cc1cc(C)on1 Cc1nc(N)c(CC(N2CCOC(CNC(C3COCCN3C)=O)C2)=O)c(O)n1 N1(C(C=CC)=O)CC2CC1(CNC(c1ccccc1OC(F)(F)F)=O)CC2 n1(CC(N2C(CN(C(C3CN(C)C(=O)N3)=O)C)CCC2)=O)ncc2ccccc12 N1(C(C(C=C)(C)CC)=O)Cc2ccc(OC)cc2CC1C(=O)OC c1(C(=O)NCC(=O)N(CCCC#C)C)occc1CNC(c1ccn(CCF)n1)=O N1(C(c2n[nH]c(C(C)(C)C)n2)C(N2CC(C)(CF)C2)=O)CCC(F)(F)CC1 N1(C(C(C)CN(C)C(c2cc(C(N)=O)[nH]n2)=O)=O)CC(=O)NC(C2CC2)C1 C1(C(=O)NCC2(CC)CCCCO2)CCCCN(C(C2(C)CC(C)=NO2)=O)C1 CN1CCn2ncc(C(=O)NC3CC(CCNC(c4ccc(C(N)=O)[nH]4)=O)C3)c21 C(=O)(NNc1nc(-c2ccccc2)cs1)c1cncc(C(c2ccccc2)=O)c1 N1(C(C2CCC(C)(C)O2)=O)CCC2(CCCC2NC(=O)C=Cc2cn[nH]c2)CC1 c1(OC)cccc(NC(C2C3CN(Cc4cccc(-c5nn[nH]n5)c4)CC23)=O)c1 O(NC(=O)C(O)CCNC(=O)CN1CCCC1C)CCCOC C1(NC(CCN(C)CC)=O)COC2(CCN(C(=O)C(F)n3ccnc3)CC2)C1 CCC(F)(F)C(=O)NC(CCNC(c1cc(-c2ccccc2)ns1)=O)C(C)C C1(C)(CNC(Cn2c(C)nnn2)=O)CCC(NC(C2CC2CN(C)C)=O)CC1 Cc1cc(N2CCC(C3CC3)C2CNC(C2CCCS2)=O)n2ncnc2n1 Cc1ccc2c(Cl)c(C(=O)NC3CC3CNC(=O)C3=CCCCC3)sc2c1 CC(C)CCCCCC(=O)NCCCC(C)NC(=O)CCc1nnc(C2CC2)o1 N1(C(CC2CCC(C)CO2)=O)CCC(NC(C2CC(=C(F)F)C2)=O)C(O)C1 c1(C(c2nnnn2C2CCCC2)(CC)NC)cnn2c1CCC2 c1(C(=O)NCC(C)(C)NC(=O)CC2CCC(=O)CC2)cc(F)cc(F)c1 c1(C(=O)NC2CCC(C)(NC(=O)Cc3nncn3C)CC2)coc(S(C)(=O)=O)c1 CC(C)C(O)C(=O)NC1CC(C)(NC(c2cnc(C(C)(F)F)s2)=O)C1 c1(C(N2C(C)(CNC(C(C)C(F)F)=O)CCC2)=O)ccc2c(c1)CCCO2 C(=O)(CCC(C)OC)NCCCN(C(CC(=O)OC)=O)Cc1ccsc1 C1(N(C(c2cc(C)cc(C)c2)=O)C)CCCC2CN(C(=O)CCC(C)(F)F)CC12 N1(C(C2C(C#N)C2)=O)CCCCC1CNC(c1cnc(S)n1C1CC1)=O N1(C(COCCCC)=O)CC(C)(CNC(C23CC2COC32CCC2)=O)CC1(C)C C1(NC(c2cncc(CNC(C34CSCC3C4)=O)c2)=O)CCc2n[nH]cc2C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC(CN(C(C(C)OCC)=O)C)(C)C N1(C(c2c(CC)nc(C)o2)=O)CC2(CC)CC1(CNC(=O)C(C)(C)C)C2 C1(C(CNC(C2(C)CCCS2)=O)OC)CCN(C(C2CCSC2)=O)CC1 O=C(CC1=CCOCC1)NCCOCCNC(=O)CC1(CO)CCOCC1 C1(NC(CNC(CC)=O)=O)CCCC1C(=O)NCC1COCC1O C(c1ccccc1Cl)=C(C)C(=O)NCC1(O)CN(C(=O)CCc2nccn2C)C1 N1(C(C2(CC)CC(F)(F)C2)=O)C2CCC(C2)C1CNC(C1CCC2CC12)=O Cn1ncc2nc(C(F)F)c(C(=O)OCCC34CC5CC(CC(C5)C3)C4)cc12 C1(CC(N2CC(NC(=O)CSCc3ccccc3)C(O)C2)=O)(CC)CCOCC1 c1(C(N2CCCC(NC(CC(=C)C)=O)C2C)=O)ccc2nnc(C(F)F)n2c1 C(c1ccc(F)cc1)=CC(=O)NCCCOCCCNC(c1cncc(O)c1)=O c1(NC(C(N2CCn3c(C)ncc3C2)=O)=O)ccc2c(c1)CCCC2=O C1(NC(C(C)C(C)(C)C)=O)CN(C(c2cc(N)cc(F)c2)=O)CC2(CC2)C1 C=C(C)C(CC(=O)N1CC(F)(C(=O)NCC(N2CCOCC2)C)C1)OCC N1(C(CN2CCC(C)CC2)=O)CCC(F)C(NC(=O)CC2CC3CCC2CC3)C1 c1(C(N2C(C)CCC(NC(=O)CCCCCN(C)C)C2)=O)cnc2ncccn12 O=C(C#CC1CCCOC1)NC1CN(C(=O)CSC(F)F)CC1F C1(NC(C(CC)SC)=O)COC2C(NC(c3ccn(C(CC)CC)n3)=O)COC12 C(=O)(N1OC2CCC1CC2)C1N(C(C(CC=C)C(C)C)=O)C2CCC1C2 c1(CC)nc(=N)[nH]c(=NCCC2(OC)CN(C(c3cccc4sccc34)=O)C2)[nH]1 N1(C(CCCOCC)=O)CCC2(CC1)COC(CNC(=O)C(C)(C)C)C2 c1(N(CCN(CCC(=O)OCC)C)C(c2ncncc2N)=O)ccc(C)c(C)c1 C(=O)(C#CC1CCCCO1)N1CCN(C(c2c(C)cc(C(N)=O)nc2)=O)CC1 O=C1CC(CC(=O)N2CCC3(CC2)CC3NC(C23CCCC2CCC3)=O)=NN1 Cc1nc2cccnn2c1C(=O)NCC(C)CN(C(=O)CCc1cc(Cl)cs1)C N=c1ccc(C(=O)NCC2CC2NC(c2csc(Br)n2)=O)n[nH]1 C(C(=O)N(C(C)CN(C)C(c1cc(C)[nH]c1C)=O)C)(C(C)O)NC(C)=O CC1(C)C(C(=O)NCC2CCC(NC(=O)COCCOCCO)C2)C1(C)C C(=O)(C(C)C(F)F)N(CC(CC)NC(C1(CN(C)CC)CCCC1)=O)CC CC1=C(C(=O)N2CC3CC3(CNC(C3C(C)(C)C3(C)C)=O)C2)CCC1 C1(NC(c2cccc(O)c2Cl)=O)CCN(C(c2cc3occc3s2)=O)CC1O CCN=C(NCC1CCC(CC(N)=O)CC1)NCC(C)C#N C1(OC)CCC2(CCN(C(c3cc(CNC(C4CC4F)=O)ccn3)=O)C2)C1 N1(C(C2C(C)(COC)C2)=O)CCCC2(C1)CN(C(=O)CCNC(=O)CO)CCO2 N1(C(C23C(C)(C)C(CC2)CC3)=O)CCC2CC(C1)CN(C(C1CCOC1)=O)C2 c1(C(C)SCC)nc(-c2cccc(C(F)(F)F)c2)n(C(c2cccc(F)c2)C)n1 c1(-c2cc(-c3n(CC(=C)C)nc(CCCC)n3)no2)ccc(OC)cc1OC C(=O)(CCN(OC)C(=O)N(C1CC(N(C)C)C1)C)NC(CC)CN(C)C Cc1cc(CCC(=O)NCC2(C(=O)NC3(C)CC3(C)C)CCCC2)n[nH]1 c1(NC(C2(O)CCN(C(C(=O)OCC)=O)CC2)=O)ccc(C(=O)NC)c(Cl)c1Cl N1(C(c2cc3n(n2)CCC3)C(=O)NCCCSC)C2CCCC1CC(=O)NC2 c1(C(=O)NCC(C(C)C)(C)NC(C2(C3CCC3)CC2)=O)ccc(Cl)c(Cl)c1O C1(C(N2CC3CC3(CNC(=O)Cn3cncc3C)C2)=O)(CC)CCOCC1 N1(C(CCC)=O)CC(O)(C(=O)NC2(C3CCCCO3)CC2)C1 Cc1ncccc1C=CC(N1CCC12CN(C(C1(C3CCC3)CC1)=O)C2)=O c1(COC)nc(C)c(C(=O)NCC2CCN2C(C2(F)CC2c2ccccc2)=O)s1 c1(C(CC)C)ccc(C(=O)NCCC2CCN(C(C3CC4(CSC4)C3)=O)C2)cc1 c1(C(=O)NC2CC(NC(c3ccnc(C)c3C)=O)C2)ccc2sccc2c1 C1(C(=O)NC2CC(CCNC(C3(F)CC3)=O)C2)CC2C=CCC(C1)C2 C(=O)(CC(C)C(=O)N1CC(NC(c2cc(Br)ccc2C)=O)C(O)C1)OC C1(CNC(C=CCNC(CN2CCC(OC)C2)=O)=O)CCC(=O)NC1C CC(Cn1cccn1)C(=O)NC1CCCC1CNC(=O)CCNC(N)=O c1(OC)ccc(C)c(OC)c1C(=O)NC1CN(C(=O)C(O)CCC(C)C)CC1O C1(C(N2C(CNC(c3c(COC)ncs3)=O)C(C)CC2)=O)Cc2ccncc2N1 O=C(N=c1cc2n([nH]1)CCCC2)NC1CSCc2ccccc21 C(CNC(=O)CCCCC#N)(C(=O)N1CC(O)CCO1)N(C)C C(=O)(CCCCNC(N)=O)NCC1C(NC(C(C)(C)C2CCCC2)=O)COC1 CCC(C(=O)N1CCN(C(=O)N=c2ccn(CCF)[nH]2)CC1C)C(C)(C)CC C(CCCC(CO)NC(C1CS(=O)(=O)C1)=O)NC(c1c(C)n(C)cn1)=O c1(C(=O)NC(C)CN(C)C(c2cncc(C#N)c2)=O)cc2ccc(Cl)cc2[nH]1 C1(C(C)NC(C2CCC(=O)O2)=O)CCN(C(C2CC2C(=O)OC(C)(C)C)=O)CC1 CC(C)(C)C(CO)C(=O)N1CC2(CCC2)CC1C(=O)NCc1csnn1 C1(C(N(C2CCN(C(c3cncn3C)=O)C2)CC)=O)(OC)CCC(C)(C)C1 c1(CSCC(=O)NCCCN(C)C(c2cccnc2)=O)ccc2ncsc2c1 C1(C(=O)OCC)C2CN(C(=O)CN(C(=O)CCC3CC3(C)C)C3CC3)CC12 CC1CN(C(=O)C=C2CCCCC2)CC1NC(c1cscn1)=O CC1=CC(C)C(c2cn(CC(F)CCNC(C3CCC3)=O)nn2)CC1 Cc1ccccc1CC1CCCN(C(=O)NCc2cn(-c3ccccc3)nn2)C1 n1(CC2CCCN(C(=O)OC(C)(C)C)C2)cnc2c1CCNC21CCOC1 c1(CNC(C(N2CCC(N(CC)CC)C2)=O)=O)cc(C)c2c(c1)CCC2 c1(C(=O)NCCCCC2CN(C(c3c(CCC)occ3)=O)C2)scc(C)c1C C(C1=CCN(C(=O)COCc2ccc(O)cc2)CC1)NC(C1C2CCCC12)=O N1(C(c2ccc(N(C)C)cc2F)=O)CC2CCC1CN2C(C1CC2C=CC1C2)=O c1(C(N2C3CN(C(C(C4CC4)OC)=O)CC2CC3)=O)c(Cl)nc2sc(C)cn12 c1(C(=O)NC23CCCN(C(c4cccc(C)n4)=O)C2C3)cc2sccc2cn1 Cc1cccc2ncnc(NC3CCN(C(=O)Cc4cc[nH]n4)C(C)C3)c12 c1(C(=O)OC)nnsc1S(=O)(=O)NNC(=O)C1CCCCN1C1CCCC1 C1(C)(CNC(c2n[nH]c(C)c2Cl)=O)CN(C(c2cccc(Cl)c2F)=O)CCO1 c1(C(=O)NC(CCCC)C(=O)NCc2ccc(O)c(C)c2)cnn2cccc2c1 c1(CC(=O)NCC(C)CNC(=O)CCNC(C2CCCO2)=O)cc(F)cc(F)c1 N1(C(C2C(CCC)C2)=O)CC(C(N2CCN(CC)CC2)=O)CC(C)(C)C1 N1(c2nc(-c3c(C)ccnc3)nc(N)c2)CCN(Cc2ccccc2)CC(O)C1 c1(C(=O)NC2CN(C(C(C(=O)OC)OC)=O)C(C)CC2)ccn2nccc2c1 C1(CCN(C(CCOCC)=O)C)CCN(C(C23CC(CC(C)C)(C2)C3)=O)CC1 O=C(C1=C(F)CN(C(c2cc[nH]c2)=O)CC1)N1CCC2(CCCC2)C1 CCC(C)(CNC(c1cccc(=O)o1)=O)C(=O)NC1(c2ncc[nH]2)CC1 C=CC1(CO)CCN(C(C23CCC(CC2NC(=O)CCC(C)C)C3)=O)CC1 c1(C(=O)NCC(C)(CO)NC(CCCC(=O)OCC)=O)cc2cccc(Cl)c2s1 C(=O)(CC1OCc2ccccc21)NCCN(CCOC)C(c1csc(CO)c1)=O C1(CCNC(Cn2c(C)nnn2)=O)CCCCN1C(=O)COC1CCOC1 C1(NC(CNC(c2cc(CC(=O)OCC)on2)=O)=O)CC(=O)NC1=O C12(CC(=O)NC3CN(C(C4CC(OC)C4)=O)CC3C)CCCN1CCC2 C1(O)(C(=O)NCC2C(NC(CSCC(C)C)=O)CCCC2)CCCC(C)CC1 CC1(C(=O)NCC2CCC(NC(c3cccc(C(N)=O)c3)=O)CC2)CCCC1O C1(NC(Cc2cn(C)nc2)=O)CCC(O)CN(C(C2(C3CCCO3)CC2)=O)C1 Cc1cc(C)c2[nH]c(C(=O)NC(C)Cc3c[nH]c4cccnc34)cc2c1 c1(NC=O)ccc(NC(=O)C(F)CC2CCCC2)cc1.c1(NCC)ccc(O)nc1 c1(C(=O)NC(CNC(CNC=O)=O)C2CC2)cccc(N2CCCCC2)c1 C(C(C)C)(C(C)C)NC(C(C)N(C(C(C)=C1CCC1)=O)C)=O C1(C)(CC)CCC(C(=O)NCC(C)(F)CNC(c2cc(C)oc2C)=O)O1 Cc1ccc(-n2cc(O)c(C(N3CC(NC(C4CC(N(C)C)C4)=O)C3)=O)n2)cc1 C(=O)(C1=NOC2COCC12)NC1C(OCC)CN(C(=O)COC(F)F)C1 CSC1=C(C(=O)NCC(C)CN(C)C(c2conc2C2CC2C)=O)CCCC1 C=C(Cl)C(C)(C)C(=O)NCC(CC(C)C)NC(c1ccc(OCC)c(OC)c1)=O C1(NC(c2cc(CO)[nH]n2)=O)CCC2CC1CN2C(c1cc2c(s1)CCOC2)=O C1(CNC(CCC(C)=O)=O)CC2(CCOCC2)CN1C(=O)C1=NOC(C)C1 N1(C(c2ncn(CC)n2)=O)CCCC(O)(CNC(C2CC2C)=O)CC1 Cc1cc(C(N2CCSCC2C(=O)Nc2cccc(F)c2O)=O)cc(C#N)c1 c1(CNC(=O)CCNCCCC)ccnc(F)c1Cl.N12CCC(C1)C2CC C(=O)(CCCCCCn1cc(C(C)(C)O)nn1)N(C(C=C)C1CC1)C Cc1cccc(C(=O)NCCC2(O)CCN(C(c3ccccc3CO)=O)C2)n1 N1(C(C(COC)C)=O)CCC(C)CC1CCNC(c1cnn(C2CC2)c1)=O N1(C(C2C(OC)CCC2)=O)CCCC(NC(c2cccs2)=O)CC1 c1(C(N2CCC(NC(C3(CC)CCNC3=O)=O)C2C)=O)nc(O)nc(O)c1OC C1(N(C(=O)CC(C)(F)F)C)CCC2CN(C(c3ccncn3)=O)CC12 c1(C(=O)NC2CC3CCC2N3C(C2CCCCC2)=O)ccc2nsnc2c1 c1(C(=O)NC(C)COC)cccnc1OCCC1CCN(C(C(=O)OCC)=O)C1 c1(C(N(C2CN(C(C(CCCC#C)C)=O)CC2O)C)=O)ccc2c(c1)nnn2C CCCCCS(=O)(=O)CC(=O)N1CCC(NC(C2(C)CNC(=O)C2)=O)C1 c1(CC)cc(C(=O)NC(C2CCOC2)CNC(C2CC(OC)C2)=O)ccc1F c1(C(=O)NC2C(NC(=O)CC34CCCC3C4)CC2)cn2cc(Cl)cnc2n1 c1(C(=O)NCCC2N(C(CCCC)=O)CCOC2)cnc2ccoc2c1 C1(NC(c2cc(O)nc(C3CC3)n2)=O)CC2CCCN(C1)C2 c1(C(N2CC3C(CNC(C(CCOC)C)=O)C3C2)=O)ccc(C(C)=O)nc1O N1(C(C(CC)OCC)=O)CCC2CN(C(c3sc4ccccc4c3C)=O)C2C1 n1(CC(=O)NCCC2(NC(CNC(=O)OCCC)=O)CC2)cc(Cl)cn1 Cc1cc(C#N)cc(C)c1NC(C1CC(F)CN1C(=O)CCC(C)C)=O Cc1nc(Cl)c(NC(=O)CC2CCCN2C(c2ncc(Br)cc2F)=O)cc1Br C1(N(C)C(c2ccnc(O)c2)=O)CC2CC1N(C(c1ncccc1F)=O)C2 C#CCC(CC(F)F)C(=O)N1CCC(CC#C)(C(=O)NCc2[nH]c(C)nc2C)C1 C1(C)(C(=O)NC2CC(CNC(c3ccc(C#C)cn3)=O)C2)CCC(C)(C)CC1 c1(C(=O)NCC2CN(C(c3n(COC)ncc3)=O)C(C)C2)c(C)nc2sccn12 CCC(C(=O)N1CCC(CC(=O)NCCc2nnc(O)o2)C1)C(C)C c1(C(N2CC3OCCN(C(C(C)OC)=O)C3C2)=O)[nH]c2c(c1C)C(=O)CCC2 C(=O)(CC1OCCc2sccc21)N(C1CN(C(=O)CCn2cccn2)C1)C c1(C(N2CCC(C(=O)NC(COCCOC)C)C2)=O)ccc(C)nn1 C1(OC)CC(NC(=O)CCSc2cccc(Cl)c2)CN(C(=O)CCCCC#N)C1 CCC(C)(C)C(O)C(=O)NC1CCC(NC(=O)C(C)(C)Nc2ccccn2)C1 N1(C(C(C)NC=O)=O)CCC(C(N2CCC(CF)C2)=O)C1 S(=O)(=O)(c1cccc(F)c1)N1CC(NC(c2cccc(NC)n2)=O)CC(F)(F)C1 C=CCCCC(C1CC1)NC(=O)CC(O)CNC(c1cnn(C)c1C)=O C(=O)(CC(CC1CC1)NC(C1CC(C)(C)C1)=O)NC(C1CC(F)(F)C1)C C(=O)(C(F)(F)C(F)(F)F)NC1CC(CNC(=O)CC2CCCC23CC3)C(O)C1 C#CC1CCC(NC(C2COC(CN(CC=CC(=O)NC)CC)C2)=O)CC1 c1(C(=O)NC2CN(C(C3C(C)C3C)=O)CC(C)C2)ccc2nn[nH]c2c1O CCCCC(O)C(=O)N1CCCC(N(C(=O)Cc2coc(C)n2)CC2CC2)C1 c1(CNC(C(C=C)O)=O)nc(CNC(c2cc(C3CC3)ccc2F)=O)cc(O)n1 Cc1nc(C(=O)NC(C2CCOC2)CNC(c2cnc(C(C)(C)C)o2)=O)c(C)s1 C1(CNC(c2ncn(C(C)C)c2)=O)C2CN(C(=O)CN(S(C)(=O)=O)C)CC12 CCCCCOCC(=O)NCCN(C(=O)C=CI)CC1CC1 CN1C(=O)CCC1CC(N1CCOC(C2CN(C(C3CCS(=O)(=O)N3)=O)C2)C1)=O C(=O)(C(F)(F)CCn1ccnn1)N1C(CNC(COCCOCC#C)=O)CC1 c1(C(N(CCC)CCNC(c2[nH]cnc2C)=O)=O)ccc(N(C)CC)cc1 C1(NC(c2cnc(C)o2)=O)CCCCC1NC(=O)C(F)(F)C1CCCC1 C1(NC(C(=O)NCC)=O)C2CN(C(=O)CCc3cnn(C)c3)CC12 N1(C(c2c(C)scc2)=O)CC(C(=O)NC2CC(C(F)(F)F)C2)CC12CCC2 N1(C(C(CN(CC)CC)F)=O)CCC(N(C)C(c2n[nH]cc2F)=O)C2(CC2)C1 C#Cc1ccc(C(=O)NC2CCC2NC(c2c(N)cccc2Cl)=O)cc1Cl C12(C(=O)NCC(CCCC)NC(c3cc(C)[nH]n3)=O)C3C4C1C1C2C3C41C#N CCC(CCC(=O)NC(CO)C(=O)N1CCCC1CC1CC1)OC Fc1cccc2[nH]c(=NCCOCC3CCCO3)nc(N3CCCCC3)c12 Cc1[nH]nc2ncnc(N3CC(=C(F)CNC(=O)C(C4CCCCCC4)O)C3)c12 C(CC(C)NC(=O)C=CCN1CCCC1)OC CCC(O)C(F)(F)C(=O)NCC1(C(C)NC(c2c(C)noc2C)=O)CC1 c12nc(-c3ccccc3)nn1CCOCCN2C.C1(OCC)CCCC(C)C1 CC1CN(C(c2ncccc2O)=O)CCC1NC(C1CC(n2ccnn2)C1)=O c1(CN2C(CNC(CNC(C3C(C)C3C)=O)=O)CC2)nc(C2CCCC2)no1 c1(CC(=O)NC2CC23CC(NC(C24CCCC(C2)OC4)=O)C3)ccc(Cl)cc1F CC#CCCCC(=O)N1CCC(NC(C2(CC)CCCCC2)=O)C1 C1(NC(CCSCC)=O)(CO)CCCN(C(C2(O)CCOC2)=O)C1 c1(C2(C(=O)Nc3cccc(C(C)=O)c3)CC2)ccc(C)cc1Cl N1(C(C(CC)N(C(=O)C(C)CC#N)C)=O)CCSCC(C)C1 CC1=C(C(=O)N2CCCC(CO)(NC(c3c[nH]c(=N)s3)=O)C2)CCCC1 c1(OC)c[nH]c(C(=O)N(C)CCOCCN(C(=O)C=C(CC)CC)C)cc1=O c1(C(=O)NCC(C)CN(C)C(c2cc(Cl)cs2)=O)cc(S(N)(=O)=O)c[nH]1 CC1CN(C(=O)CC(C)(C)c2ccccc2)CCC1NC(C1CC12CCC2)=O c1(C(N2C(C)CC(NC(C(C)N3CCC3)=O)C2)=O)cnc(O)nc1O C(CCCCC(=O)N1CCC(c2cn(CCC(C)C)nn2)C1)c1c(C)cccc1 c1(C(=O)OC)c(C)cc(C)nc1N1C2CCC1(CNC(=O)CC1(O)CCC1)CC2 CC(O)CC(C)(C)CNC(C1(CNC(=O)CCC2OCCO2)CC1)=O C1(NC(CCC(=O)OCC)=O)CS(=O)(=O)CC1NC(=O)CCc1ccc(O)nn1 N1(C(CN2C(C)CCC2)=O)CC2(CCC2NC(C2CCC(N(C)C)CC2)=O)C1 CC1CCN(C(c2csc(-c3cnn(C)c3)n2)=O)C(CNC(C2CCCO2)=O)C1 CC(C)C(C)C(C(=O)NCC(C1CC1)NC(c1ncc[nH]1)=O)NC(=O)OC(C)(C)C C1(C(N)=O)CCN(C(=O)C(Cc2ccccc2)NC(=O)COCCCF)C1 n1(CC2(OC)CCC2)c(N(C)CCCc2cccs2)nnc1-c1cccc(C)n1.OBr c1(OC)cccc(F)c1CNC1CC1C(=O)Nc1ccc(Cl)cc1O CC1(O)CCCC1NC(c1ccc(CNC(C2(n3nccn3)CC2)=O)cc1)=O c1(C(=O)NC(C(N2CCCC(C)(O)C2)=O)CCF)cncc2[nH]ccc12 C12(C(N(CCNC(=O)Cc3c(C)cccc3Cl)CC)=O)CCC(CF)(CC1)CC2 C(C(CNC(=O)Cc1ccccc1F)C(F)(F)F)NC(c1c(=N)[nH]cnc1)=O Cc1cc(C(C)C(N2CCCC(CNC(=O)C#CC(=O)N(C)C)C2)=O)cc(F)c1 C1(C)(NC(CCC2CCN(C(C(C(C)C)C)=O)C2)=O)CC2(CCC2)C1 Cc1[nH]c(C#N)cc1C(N1CC2CC1C2C(=O)NCC(O)CC1CCC1)=O CC1CN(C(=O)C=Cc2nccs2)CCC1C(=O)NC1CCC2(CC1)N=N2 c1(C(N2CCC(F)(CNc3ncc(F)cn3)C2)=O)cc(Br)c2cc[nH]c2c1 C#Cc1ccc(C(=O)NCC(C(=O)NCc2cc(Cl)ccc2O)N(C)C)cc1 c1(OC)cccc2cccc(C(=O)NCCCCNC(C3(F)CCCC3)=O)c12 c1(C(=O)NCC23CC2CN(C(=O)C=Cc2cccs2)C3)coc2ccccc12 N(C)(C(=NCCc1ccc(Cl)s1)NC1CCS(=O)(=O)C1)C(C1CN(C)CCO1)C O=C(C1=NOC2COCC12)NCC1(O)CCCN(C(=O)Cc2ccoc2)C1 c1(C(=O)NCC2CCN2C(c2ccc([N+](=O)[O-])s2)=O)ccn2c1CS(=O)(=O)CC2 N1(C(C)CCNC(=O)OC(C)(C)C)CCSC2(CCCCC2)C1 c1(CC(N)=O)n[nH]c2ccc(F)cc12.c12cccc(c1)OC(=O)CCC2 C1(NC(c2onc(C(C)(C)C)n2)=O)CC2CC1CN(C(=O)C(C)(F)F)C2 C1(CNC(c2cnc(CC)s2)=O)C2CC1N(C(=O)C=CC1CCCO1)C2 C=CCC(CC)C(=O)N1CCN(C(c2nn[nH]c2Cl)=O)CC1CO C1(CC(N2C(CCNC(C(C3CC3)OCC)=O)CCC2)=O)CCC(C)CC1 C(C)(C)(C(C)CC(=O)NC1CN(C)CC12CC2)NC(c1n(CCC)ccc1)=O c1(C(=O)NCC2CN(C(C3OCCC(C)C3)=O)C2)ncn2cc(Cl)ccc12 c1(CNc2ccc(C(=O)Nc3c(NC=O)cccc3)nc2)cccc2c1OCO2 C1(N(C(CC)=O)C)CS(=O)(=O)C12CCN(C(c1ccc(P(C)(C)=O)o1)=O)CC2 N1(C(c2ncnc(OC)c2F)=O)CCCC2(CCN(C(=O)C(OC)OC)C2)C1 c1(C(=O)NCCC2(NC(CCCc3scc(C)n3)=O)CC2)noc2c1COCC2 c1(CC(=O)NC2C(NC(c3n(C)cnc3)=O)CCCCC2)ccc(S(C)=O)cc1 c1(NC(C(CC)C(C)O)=O)ccc(OCCN(C)C)c2cccnc12 N1(C(C2CCC(C)C2)=O)CC2(NC(=O)CCCC3CCCC3)CC1C2 N1(C(C(C)=CC2CC2)=O)CCC2(CCCN2C(c2ccc(N)c(Cl)c2O)=O)C1 C1(C(=O)OC)CC(C2(NC(c3cnc4n3CCS4)=O)CC2)C1 C(=O)(C(C)C(O)C(C)C)NCCC1CC(C(=O)NC(COCC)CO)C1 N1(C(CN(C)C2CC2)=O)CC(CCO)C2(C1)CN(Cc1ccc3ncsc3c1)C2 C(=O)(C1=C(Cl)CCC1)NC1C2CN(C(C3(CC#C)CCCCO3)=O)C1C2 C1(C(=O)NC2(C)CC(NC(C3CC(F)(F)C3)=O)C2)CC2CCC(C1)N2C1CC1 c1(OC)c(CC(=O)NCCCNC(c2cccc(OC)c2)=O)cccc1C#N c1(OC(CNC(c2cn(C(C)C)nc2)=O)C)cc(F)cc(F)c1 c1(C(N2CC(NC(c3c(OC)csc3)=O)C(C)C2)=O)cc(OC)cc(Cl)c1O C(=O)(CS(=O)(=O)N(C(c1ncc[nH]1)C1CC1)C1CC1)N(CC(N1CCC(C2CC2)C1)=O)C C1(CN(C(CC2(CC)CC2)=O)C)COCCN1C(C1C=CCCC1)=O N1(C(CC(CC)C2CC2)=O)CCCC(O)(c2cn(CCN(C)C)nn2)CC1 CCCC(C)C(=O)N1CCCC1CCCNC(=O)C(C)(C)n1ccnn1 C1(NC(CCOCCOC)=O)CC2CC(NC(c3cc(OC)nc(Cl)c3)=O)CC12 c1(C(N(CCC(=O)NCC2CC2CO)CCC)=O)ccc(Cl)s1 c1(CC)ncccc1C(c1nnnn1CC(F)F)NCc1ccnn1COC CC(CC(=O)N1CC2CC1C2NC(C1(N(C)C)CCCSC1)=O)P(C)(C)=O CC1CCC(C(N2CCCC2CN=[N+]=[N-])=O)N1C(=O)CN1CCCC1 N1(C(c2cc(C)c(O)cc2)=O)CCn2ncc(CNC(=O)CC3CCC4CC34)c2C1 Cc1oc(C)c(C(=O)NCC2CCCC2C(=O)Nc2ccc(Cl)cc2)c1C N1(C(C2(CCN(C)C)CC2)=O)CCC2(CCC(NC(=O)C#CC3CCOC3)C2)C1 c1(CC(C)NC(CC=C)C2CC2)nnnn1C1CCCCC1 c1(N2CC3(C(NC(c4c(C)cn(C)c4)=O)CCS3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl N1(C(C2OCCN(C)C2)=O)CC2CCN(C(c3cnc(C4CC4)nc3O)=O)C2C1 C1(CNC(CC(C)OC)=O)CC2(C1)CN(C(=O)C(C)n1cnnn1)C2 C1(NC(C2C(C#C)C2)=O)CCCCN(C(c2cn(-c3ccccc3)cn2)=O)C1 CCC(CCOC)C(=O)N1CC(F)CC1CNC(=O)Cc1cc(OC)no1 O=C1CC2(CCN(C(C34CC3CN(C(=O)CC3CCCCO3)C4)=O)CC2)N1 N1(C(C2C(CNC(=O)CC3COCCO3)CCO2)=O)CC2CCC2C1 C1(C(=O)NCC(N2CC(CC(C)NC(CC=CC=C)=O)C2)=O)C=CC=CC=C1 CCCC(F)C(=O)NCC1(CNC(c2cnn(C(C)C)c2)=O)CC12CCC2 C1(CC(=O)NC2CCC(CNC(C(C)c3cccs3)=O)C2)CCC2(CCC2)O1 Cc1ccccc1OCCC(=O)NCC1CC(C)N(C(=O)CO)C1 CCCC(C)CCN1CCC(N(C(=O)C=CC=C(Cl)Cl)CC)C1 N1(C(c2cc(N)c(F)cc2)=O)C2CCC1CN(C(=O)Cc1cc(F)cc(F)c1)C2 N1(C(CC(CCCCC)C)=O)Cc2ccccc2CC1CNC(=O)C(=O)NCC n1(CCOC)cc(C(=O)N(CC(C)O)CCNC(=O)CSCC(N)=O)cn1 c1(CC)nc(C)[nH]c1C(N1CCC(=CCNC(=O)C(C)CC2CCC2)CC1)=O C1(C)(CCOC)CN(C(C2CC(N)CC(F)C2)=O)CCO1 Cc1nn(C)c(Br)c1C(N1CC(NC(=O)CC2CC3(CC3)C2)C1)=O.C(C)(C)(C)OC c1(C(N(CCCNC(C(C(C)C)OC)=O)C2CC2)=O)cc(N)cc(F)c1 c1(C(=O)N(CCCF)C)cc(N(C)C)cc(F)c1 CCC(C(=O)N1CCCC1CC(=O)N(CCOC)Cc1nc(C)no1)N(C)C.CSC N1(C(C2N(C(CCCSC(C)(C)C)=O)CCC2(C)C)=O)CCC12CCC(O)CC2 C#CCN(OC)C(=O)C1(CF)CCN(C(C2Cc3nccn3C2)=O)C1 N1(C(C2C(C)(N(C)C)C2)=O)CC(SC(F)F)C2CCCC12 N1(C(Cc2c(C)ncs2)=O)CC(CNC(C2(CF)CC(F)(F)C2)=O)CCC1C [N-]=[N+]=NCC(C(=O)NC1CCCN(O)C1=O)NC(C1CC1(F)Cl)=O N1(C(C(CC)F)=O)CCC2(CC1)CC2(CO)CNC(=O)CCc1nccn1C CCCCCCC(C)C(=O)NC(C)CCNC(=O)CC1CC2CCC(C1)N2C N1(C(c2c(COC)cco2)=O)CCC(NC(C2(C3CC3)CC2)=O)C(C)C1 C(CC(C)(C)C(=O)N(C1CCC1)CCO)NC(C(C)n1cncn1)=O C=CCC(C(=O)N(C(C)CNC(=O)CC1C=CS(=O)(=O)C1)C)NC(C)=O C1(CNC(=O)NC(c2nn[nH]n2)c2cccs2)C=CCN(Cc2ccccc2)C1 Cc1sc(C(=O)NCC2CCC23CN(C(=O)CCC#N)C3)c(C)c1Br C(=O)(CC(CC)CCCC)NCC(C(=O)NC(C#C)(C)C1CCCC1)C(C)(C)C C1(C(C)C)CN(C(c2ccnn2CC#N)=O)CCN1C(=O)CCCc1ncco1 CCCCC(C)C(=O)N1CCC(C)(CNC(C2CCNC(=O)C2)=O)C1 N1(C(C(C)N(CC)CC)=O)CC(NC(=O)C(CC)CCC)C2(CCCC2)C1 C(=O)(CCCC(=O)C(=O)CO)NC(C(C)c1ccco1)=O.c1(N)ccccc1C#N c1(C(=O)NC2(C)CCC(NC(=O)C3=CCS(=O)(=O)C3)CC2)cccn2nccc12 C1(NC(C2(OCC)CCOC2)=O)CCCC(NC(=O)CC2CC2CC)C1 c1(C(N(CCCN(C(C(CC)(C)CO)=O)C)C)=O)cc2c(Br)cccn2n1 c1(OC)ccnc(C(N2CC3CC2C3NC(C2CC2C)=O)=O)c1 C1(CC(=O)NCC(CNC(c2csc(C)c2C2CC2)=O)C)CC2(CCCC2)CO1 C=C(Cl)CC(C(=O)N1CC(c2noc(C)n2)C1)NC(c1cn(C)nc1CC)=O C1(C)(NC(C(c2ccccc2)OC)=O)CC(NC(C2CC2(C)C)=O)C1 C(=O)(C(C)(O)C(C)C)NCCC1CC(NC(Cc2c(C)ccnc2)=O)C1 C1(NC(C(C)S)c2nnnn2CCOCC2CCCCC2)C2CCC(F)(F)C12 C1(CC(C)C)C(=O)N(C2CCC(c3ccccc3)C2)C(=O)N1C n1(CC(=O)NC2C(NC(COCCCC#C)=O)C2)c(C)cc(C)nc1=O Cc1cc(Cl)c(C(=O)NCc2cn(CCNC(=O)CCC3(C)CC3)nn2)cc1F c1(SCCOC)ccc(NC(C(=O)NC(=O)C(c2ncccc2C)N)=O)cc1 c1(OC)cc(N)c(C(=O)NCC2(F)CCC(CNC(C3CCCC3)=O)C2)cc1F c1(C(=O)NCC2(CNC(C(F)=C(C)C)=O)CCCC2)ccc(F)cc1N N1(C(C2(C=C)CCC2)=O)CCN2C(=O)C(CCC)CC2C1.C1CC(=O)NC(=O)N1 N1(C(c2c(C)noc2N)=O)CCC2C(NC(c3cnn(CC(C)C)c3)=O)C2CC1 N1(C(CCC#CC)=O)CC2CCN(C(c3c[nH]nc3OCC)=O)C2C1 c1(-n2c(C3CC3C(C)C)nc(C(CC)O)n2)nc2ccc(C)cc2[nH]1 CC1(NC(=O)C(F)=C2CCCC2)CN(C(C2CCCC2O)=O)C1 C(=O)(C1=C(Cl)CCOC1)NCC1(F)CN(C(c2ccc(CS(C)(=O)=O)o2)=O)C1 c1(C(N(C2CCCN(c3ccncn3)CC2)C)=O)cncc(Cl)c1Cl c1(C(N(CC(=O)NCC(CC=C)OC)C)=O)c(C)cc(Br)cc1Cl CN1CCN(C(c2cc(O)ncn2)=O)CC1C(=O)NC1CCN(CC2CC2)C1 C=CCC(C)(C)C(=O)NCC(C)N(C)C(c1cccc(-c2ccco2)c1)=O N(C(=NCC1(CO)CC12CCC2)NC(C)C)C(C#C)Cc1ccc(Cl)cc1 N#Cc1cc(CC(=O)NC(Cc2ccc(Cl)cc2)C(=O)O)cc(Br)c1 C1(CNC(c2c(C(C)(C)C)ocn2)=O)CCCCN(C(C2CNC(=O)N2)=O)C1 c1(C(=O)NC(CNC(c2ccnc(C)n2)=O)C2CCC2)ccc(N)c([N+](=O)[O-])c1 N1(C(C)=O)CC(NC(c2cc(S(=O)(=O)N(C)C)c(Cl)cc2Cl)=O)CC12CCCOC2 c1(N(C(=O)NCCCc2ccc(C)s2)C(C)C)ccc(Cl)c(C(F)(F)F)c1 c1(NC(C(C)SCC(=O)Oc2cccc(C)c2)=O)ccc(-n2cncn2)c(C)c1 C1(C(=O)NCCC2(COC)CC2)CC(=O)CN1C(=O)C(C1CCCCC1)=O Cc1ccc(C(N2CC(O)(C(C)NC(C3CCS(=O)(=O)C3)=O)C2)=O)nc1C C1(Nc2cccc(C(C(C)C(F)F)=O)c2)CCCN(C(=O)OC(C)(C)C)C1(C)C c1(C(=O)NC(C)C(C)(C)NC(=O)CC2CC2(C)C)ccc(C(N)=O)nc1 C(=O)(C(C)(C)C(O)C(C)C)N(Cc1c(C(N2C3CC(=C)CC2CC3)=O)occ1)CC Cc1ccc(C(N2CCCC2C(C)NC(c2ccn(C(F)(F)F)n2)=O)=O)o1 n1(CCC=C)c2nnc1C(OC)C1CCN2C1.c1(COC)ccc(Br)s1 CC1CCCCN1CC(=O)N(C1CCN(C(=O)CCCO)C1)C C1(C(=O)NCCOC)CN(C(=O)OC(C)(C)C)C2CC12.c12cc([nH]n1)N2 c1(CC)ccc(F)c(C(N2CC(NC(=O)C(C)NC(C)(C)CC)C2)=O)c1 Cc1cccnc1C(=O)NC1CCCC1C(=O)NC(C)C(C)(C)C C=C(C)CC(C)C(=O)N(C1CCC(NC(=O)Cn2ccc(C3CC3)n2)CC1)C c1(CCC(=O)NCC=CCNC(CC2(C)CCCO2)=O)nc2cccnc2[nH]1 N1(c2n(C)nnn2)CC2(CCC(CNC(c3cn(C(C)(C)C)cn3)=O)O2)C1 C(C)(CCC(=O)NC(CCC1CC1)C(=O)N(C1CCN(C)CC1)C)OCC c1(C(CNC(c2ccoc2Br)=O)(F)F)cccc(Br)n1 CCC(CC(F)(F)F)C(=O)N1CCN(c2nc(C3CC3)nc(=N)[nH]2)CC(O)C1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NC1C(C)CCN(C(=O)C2=CCCC2)C1 C1(F)(CC(=O)NCCCN(C(C2C(C=C)C2)=O)C)CN(C(=O)OC(C)(C)C)C1 CC1C(NC(C2OC(C)CC2C)=O)CC2CCC1N2C(=O)C1=CC2CCCC12 CCCCC(C(=O)NCC1(C(C)(C)O)CN(C(c2sc(SC)cc2C)=O)C1)N(C)C C1(C(N(CCOC)CCNC(=O)Cn2cc(N)cn2)=O)CCC2(CCCC2)CC1 C1(NC(C2N(C(c3n(C(C)C)ncn3)=O)CCC2)=O)CCN(C)C(=O)C1 C1(C(N(CCN(C(C=C(C)C(F)F)=O)C)C)=O)CC(=O)N(Cc2ccccc2)C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC1CNC(=O)Cc1cnsc1 CC(CC(F)F)C(=O)N(C(c1ccccc1)CNC(c1ccc(F)cc1O)=O)C C1(NC(C(C)N2CCC2)=O)CN(C(=O)C=C2CCCC2)CC12CCC2 C1(C(=O)NCCn2c(CC)ncc2)N(C(=O)COC(C)(C)C)CC12CCCC2 C(C(=O)N(C(CNC(=O)CN(C)C)C1CC1)C)NC(C)=O.C(C)(C)(C)O c12cc(ncn1)S2.c1(CN(NC(NCc2ccccc2)=S)CC)ccc(Cl)cc1 C(C(C)(C)CC(=O)N1CCC(NC(N)=O)CC1)NC(c1c(OC)cncn1)=O CN(C)N1CCCC1C(=O)NC1CCOCC1C(=O)NC1CC2C=CC1C2 C1(C)CCN(C(=O)CCC2(C)CC2)CC1(C)C.CCCCCCOCC.C1(C)C(=O)N1 C1(NC(c2cnc(CC)s2)=O)CCC12CN(C(=O)C(=O)Nc1ccccc1)C2 c1(C(=O)NC2CC3C(NC(Cn4cc(C(C)O)nn4)=O)C3C2)cncn(C)c1=O C1(C(=O)NCCC(C)NC(C2C3COCC23)=O)CC2(C1)CC2F CC1CCCCC1(CNC(c1cc(C#N)c[nH]1)=O)NC(C1CC12CC2)=O Cc1cccc2c1OCC2C(=O)NCCCNC(c1ncc(F)cc1N)=O N1(C(c2cnc(Cl)s2)C(=O)NCc2cccc(OC)c2)CCc2scc(Br)c2C1 N1(C(c2c(OCC)cccc2)=O)CC2(CCC2NC(=O)CC(C)C(F)F)C1 C(=O)(C#CC1CCCCO1)N(C1CN(C(c2cc(OC)c(O)cc2)=O)C1)C CC1(C)CCN(C(=O)CC2CC3(CCC3)C2)CC1C(=O)NC(CCO)C(F)(F)F CCC(C)(COC)C(=O)NC1C=CC(C(N2CCC(C)(F)CC2)=O)C1 c1(C(=O)NCC(C)(C2CC2)NC(C(COC)N(C)C)=O)c(F)ccc(F)c1Cl C1(C(C)(C)C)CCCCN(C(=N)NCC(O)Cc2ccc3c(c2)OCCO3)C1 CC1CC(C(F)(F)F)CC(C)N1C(c1nnsc1N)=O c1(C(c2nnnn2C(C)C)NCc2ccc(C)o2)c(Br)cnc(Cl)c1F Cc1ccnc(C(=O)NC2CCCN(C(=O)CC3CCCO3)C2)c1O CCS(=O)(=O)c1ccc(C(=O)NC(C)C(C)NC(=O)CCN(C)CCO)c(N)c1 C1(N(CCCN(C)C(c2cn(C)nc2C(N)=O)=O)C)CC2CCCCC2NC1=O C1(C(N(CCNC(CC(CC)SC)=O)C2CC2)=O)COC(C)(C)CO1 C(CC(F)F)(C(=O)NCCn1cnnc1)NC(COCCCOC)=O c1(C(=O)NC(CNC(C(COC)(C)OC)=O)(C)C)cccc2c1ncn2C C1(NC(C(C)OCCC#C)=O)CC12CCC(NC(c1cnn[nH]1)=O)CC2 C1(CC)(NC(=O)CCc2nc(C3CC3)no2)CCCN(C(=O)CCCF)C1 N(C1CN(C(C23CCCN(CCC2)C3)=O)CCc2ccccc21)C(C(C)SC)=O CCC(C)(C)C(O)C(=O)NCC(c1ccccc1Cl)OC(F)F N1(C(C(C)OCCCCCC)=O)CC(NC(=O)COCCc2cccs2)C(C)C1 C(CCCCC(=O)N(CC(C)C(=O)NCc1ccc(Cl)o1)C)SC N1(C(C2(C#C)CCCC2)=O)CCC2(CC1)CC(CNC(c1c(C)csc1Cl)=O)C2 N1(C(C2CC(CC)C2)=O)CC(N(C(=O)Cc2ccc(Br)cc2)C)C(F)C1 c1(C(=O)Nc2c(F)cccc2[N+](=O)[O-])cn2c(n1)CN(C(=O)NCCCCl)CC2 CC(CN(C)C(c1cn2c(n1)CCC2)=O)N=c1nc(C2CCCCC2)[nH]s1 C1(N(C)C(c2c[nH]nc2OCC(F)F)=O)CCCN(C(c2ccn(C)c2)=O)C1 Cc1cc(N2CCN(C(=O)C(c3ccc(F)c(F)c3)C)CC2C)ncc1C#N C1(C(NOCC(=O)OC)=O)CN(C(=O)C2=CCCSC2)CC12CCC2 C#CC1CN(C(c2cccc(O)n2)=O)CCN1C(c1cnc(O)c(F)c1)=O N1(C(c2c(C)nn[nH]2)=O)C2CCCC1CC(NC(=O)Cn1nc(O)ccc1=O)C2 C1(C(=O)NCC(C)(C)NC(CNC(c2cccc(C)c2)=O)=O)CCCC2(CC2)C1 N1(C(C2(C(=O)OCC)CCC2)=O)CC2(CCCC2NC(c2cncc(Cl)c2)=O)C1 CC(C)C(CN=C(NC1CCC1)NCC1CCS(=O)(=O)C(C)C1)C=O.C1(CC(C)C(=O)OC)CC1 CC(O)C(C)C(=O)NCC1CCCC1NC(c1cc(C2CC2)[nH]c1C1CC1)=O C1(C(=O)NCC(CC(=O)NCC(=O)NCC=C)OC)CCCCC1(C)C C1(=O)C2=CCN(C2)C(=O)OCNC2CN1C(C)CN2C.C(C)(C)(C)OCC Cn1cc(C(=O)NCC2CCC2NC(=O)C=Cc2cncs2)c2cccnc12 c1(C(N(C(C)CN(C(=O)COC(F)(F)F)C)C)=O)cc(C)n(-c2cnn(C)c2)n1 C12(NC(c3scc(C)c3)=O)CCCN(C(=O)C(O)CC3CCCCC3)CC1C2 c1(C(=O)NCCNC(c2cnn(C3CC3(F)F)c2)=O)ccc2c(c1)CCCS2 c1(C(=O)NC2(CNC(C(C(C)C)SC)=O)CCOC2)cc2c(cn1)NC(=O)CO2 CC(C)C(C)(O)CNC(C1(NC(=O)CC2CCCNC2=O)CC(F)C1)=O C1(CC(=O)NC)CN(C(=O)C(C)(C)c2ccno2)CCN1C(C1CC=CC1)=O n1(-c2c(C)cccc2)nc(C(=O)N(CCNN2CCCC2)C2CC2)c2c1CCC2 CC1(C)CN(C(=O)C2=CCSC2)CC1CNC(c1cn(C2CC2)nn1)=O [N-]=[N+]=NCCCCN(C(c1nnnn1C1COC1)C1CC1C1OCCO1)C1CC1 c1(C(=O)OC)ccc(C(C)CC2N(C(OC(F)F)=O)CCC2)cc1Cl CC(CCNC(=O)COc1ccc(F)cn1)CCNC(c1cnn(C)c1N)=O C1(NC(C2C(c3cn(C(C)C)nc3)C2)=O)CN(C(=O)Cc2csc(Cl)c2)CC1O N1(C(C23OCC(C)(C2)C3)=O)CC(NC(c2cnc(S)nc2)=O)C(S(C)(=O)=O)C1 C(=O)(CC(C)(F)F)N1CC(OCCNC(CCc2c(C)ncs2)=O)C1 C1(C)(CNC(C(CC2CCC2)NC(Cc2ccn(CC)n2)=O)=O)NC(=O)NC1=O C1(CNC(C(CCC)O)=O)CN(C(c2cnc(C)nc2C)=O)C(C)(C)C1 CC1C(C)N(C)CCN1C(C1(NC(=O)CN2CC(C)(C)C2)CC(O)C1)=O c1(C(=O)OC(C2CCCN(CC)C2)C#C)cccn2ccnc12 c1(CC(=O)NC2C(C)(C)CN(C(=O)C=CC3CCCC3)C2)c[nH]c2ccccc12 C(=O)(C(CC=C)CC(C)C)NC(CC#C)(C)C(=O)NCCCN(C)C1CC1 CCC(C)(CNC(=O)C=Cc1cncn1C)C(=O)NC1CC(C)(C(N)=O)C1 C(c1cncn1C)=CC(=O)NC(C1CCCC1)CNC(c1n(CCC)ncc1)=O C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CN(C(C2CCNC2=O)=O)CC12CC2 N1(C(C(F)=C(C)C)=O)CCCCC(CNC(c2c[nH]cc2C(C)(C)C)=O)C1 CCC(C(=O)NCC(CC(=O)NCCc1cn[nH]c1)OC)C(C)(C)CC Cc1cc(CCC(=O)NCC2CCCCC2NC(C2CS(=O)(=O)C2)=O)cc(C)c1 C1(NC(C2ON=C(C(C)C)C2)=O)C(C)(C)CN(C(C2CCCCC2)=O)CC1(C)C c1(C(=O)NC2CC(NC(CN(C(C)C)C)=O)C23CCC3)cc(O)cc(C#N)c1 C=CC(C)(CC)C(=O)N(C(=O)CN1CC(O)C1)C(C)(C)C N1(c2c(C)c(NC(=O)C(C)CN3CCCCC3)ncn2)CCn2c(cnc2C)C1 C1(C(N2CCC(CNC(C3(CC#C)CC3)=O)CC2)=O)CN(S(=O)(=O)N(C)C)C1 c1(C(N2CCC(CN(C(C(C)SC)=O)C)C2)=O)cn(C)cc(Br)c1=O c1(OC)cccc(C(=O)NC2CC(NC(=O)C(C)c3ccsc3)C(O)C2)n1 CCCCN=C(NCc1cc(C)co1)N1CCC(NC(=O)NC)C1 CCCC(CC(=O)N(C)CC1COCCO1)NC(C1CC2CCC(C1)O2)=O C1(C(=O)NCCCN(C(CC=CC=C)=O)C2CC2)CCc2nc(C)sc2C1 n1(CC)nc(C(=O)NCC2COCC2NC(=O)COC(C)(C)C)c2c1CCOC2 c1(NC(c2c(NC(C(OC)OC)=O)cnc(Cl)c2)=O)cc(F)c(F)c(F)c1 c1(C(=O)NC(C)CNC(C2(c3cccnc3)CCCC2)=O)ccc(CO)cn1 C1(NC(CSCCN(C)C)=O)CN(C(=O)Cc2csc(-c3ccoc3)n2)CC1O c1(SC)cc(C(=O)NC23CC2CN(C(c2cn(C4CC4)nn2)=O)C3)ccn1 C1(CC(N2C(C)CC2C(=O)NCC2(C(=O)OC)CC2)=O)CCCC2CC12 C(CC(C(C)(C)C)NC(c1cc(Cl)ccc1Cl)=O)N(C(=O)CNC=O)C CC1(C)CC(NC(=O)CC2CCCCCCC2)CN1C(=O)C=CC1CC1 c1(C(=O)NCC(C2CCCCC2)NC(c2sccc2F)=O)cc2ccccc2o1 C1(C)(COC)CC(NC(c2cc(Cl)cn2C)=O)CN1C(c1csc(C)n1)=O N1(C(CC2(C#C)CC2)=O)CCN(C(C2COC(C)C2)=O)C(CCC)C1 N1(C(Cn2c(C)csc2=O)=O)CCC2CN(C(=O)C(c3ccnn3C)C)CCC12 CN1CCC(C(=O)NCc2cnn(C)c2C(=O)NC23CCCCC2C3)CC1=O c1(C(=O)NC(CC)CN(C(=O)CC#N)C)cnn(C)c1-c1ccccc1 CC1(C)CN(C(c2ccno2)=O)CCC1NC(=O)CSCc1ccccc1 C(=O)(C=C1SCC(=O)N1C)NO.N12CCC(C(O)C1)n1cc2nn1.c1(C(=O)NCOCF)ccccc1.C(C)C CC1CCOC(C(=O)NCc2occc2C(N2CCCC(C)C2)=O)C1 C(=O)(NN1CCN(C2CCCC2)C1=O)N1CCCC(C(C)C)(CO)C1 C=Cc1cnn(C)c1C(=O)NC(C1CCCCN1C(c1cc(Cl)cnn1)=O)C C(=O)(C(C(C)C)NC(=O)CSCCC#N)N1C(C)(CCC)CC1 N1(C(CCc2cc(C)[nH]n2)=O)CCC2C(NC(=O)C(C)Cc3ccccn3)CC12 C12(NC(c3c(CC)ocn3)=O)CC(CNC(=O)C(=O)N(C)C)(C1)OC2C C(c1cncc(C)c1)=CC(=O)NC(CC)CNC(c1cc(Br)ccn1)=O c1(CNC(c2c(C)noc2)=O)ccc(CNC(C2CCSC(C)C2)=O)cc1 C(=O)(C1=COCCC1)NCC1CN2CCC1CC2.c12ccc(s1)C(=O)NC(=O)C2 c1(NC2(CO)CN(CCO)C2)cc(O)ncn1 C(CC(=O)Nn1cccn1)N(CCOC)C(C1CC1(F)Cl)=O C1(C(C)C)C(NC(=O)C(Cl)=CCl)CCN1C(=O)CC1CC2(CCC2)C1 Cc1c(C(=O)NCC2(O)CCN(C(=O)CCc3nncs3)C2)ccc2c1CCC2 c1(CC)ncc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)C(O)P(C)(C)=O)n1 c1(C(=O)NC2CN(C(C(CCC)C)=O)CC2O)occ2c1CCCC2 c1(OC)ccc(C(=O)NCC2CN(Cc3cc(Br)c(Br)s3)CCO2)cc1 N(C1CCCc2ccc(Br)cc21)c1cccc(S(=O)(=O)NC2CCSC2)n1 N(C1c2ccccc2OCC1F)C(C(=O)NCCc1cc(Br)cc2c1OCC2)=O c1(C(=O)NCC2CCCN(C(CC(CC)CC)=O)C2)cc2nc(OC)ccc2[nH]1 c1(N(C2CCN(C(c3ccc4cnnn4c3)=O)C2)C)cc(S(C)(=O)=O)ncn1 c1(CCC(=O)NC2CC2CNC(c2nocc2C2CC2)=O)nncnc1O CC1(C(=O)NCC2CC(NC(c3cnsn3)=O)CCO2)COC(=O)OC1 c1(C(=O)NC2CCC=CCC2)cccc2[nH]ccc12.CC12CC(C1)C(=O)NC2 c1(C(=O)NCC(C2CC2)NC(CC(c2c(C)cccc2)C)=O)cnc(F)c(F)c1 CN1CCC(C(=O)NC2CCC2NC(c2cc3n(n2)CCC3)=O)c2ccccc21 c1(C(=O)Nc2cc(C)c(-n3cccc3)cc2)cccc2c1CC(=O)N2C C1(NC(C(C)(C)OC(C)=O)=O)CCN(C(=O)Cn2cnnc2O)CC1C(N)=O n1(CCOC)cccc(C(N2CCC(NC(c3cnn4ccsc34)=O)C2)=O)c1=O Cn1cc2c(n1)CC(C(=O)NC1CCN(C(C3CCS(=O)(=O)N3)=O)C1)CC2 N1(C(c2c(C)nsc2C)=O)CC(C(=O)NCc2ccco2)C2(CC2)C1 N1(C(=O)NCc2ccc(Cl)s2)CCn2ncc(-c3ccnnc3)c2C1 C1(CC)(NC(C2CC(C)(C)C2)=O)CCCN(C(c2ccc(C(C)=O)s2)=O)C1 c1(N)ccc2c(n1)OCCO2.C12(OC)CCC(CO)(CC1)CC2.C1CC(=O)N1 CCC(C)CCC(O)CC(=O)NC(C1CCN(C(c2cc(CO)oc2C)=O)C1)C c1(C(N2C(C)CN(C(c3cnccc3Br)=O)CC2)=O)cccc2nc(O)oc12 CC(CC(=O)NCC(C)(C)CNC(=O)CCCNC(N)=O)n1cccc1 CC1CN(C(c2ccc3c(c2)COC3)=O)CC(C)C1NC(=O)C(Cl)=CCl C1(C(=O)NCCN(C(=O)C=Cc2nnc(C(C)C)o2)C2CC2)(OC)CCC12CCC2 CC1(C)CN(C(c2cc(N)c(N)cc2F)=O)C(C)(C)C1O c1(C(=O)NC(C)CNC(C2(CF)CC2(F)F)=O)ccc2c(c1)nc(O)n2C CCC(CC(=O)N1CCC(F)(C(=O)NCCC2CCCC23CC3)C1)CC(C)C C1(CC#C)(NC(C2C3CC(NC(=O)CCC=C)CC32)=O)CCCCC1 C=C1CCC1(C(=O)NC1CCC(CCNC(=O)CCNC(C)=O)C1)C(=O)OC c1(CC)ccc(F)c(C(=O)NC2(CNC(=O)C=Cc3ccncn3)CC2)c1F Cc1[nH]nc(C(=O)NC2CCCC2NC(=O)CCCCc2ccccc2O)c1O Cc1occc1CC1CC1C(=O)NC12CC(NC(C3(c4ccccc4)CC3)=O)(C1)C2 c1(C(=O)NC(CNC(Cn2ncc(C#C)c2)=O)C(C)C)c(C)ccc(C)c1C c1(C(=O)NC2C=CCN(C(CCC3(C)N=N3)=O)C2)nc(C)ncc1Cl Cc1cccc(CNC(N2CCCCC2C(C)O)=O)c1-n1cccn1 C(C(CN=c1[nH]c2c(c(=NCCC(C)c3cn[nH]c3)[nH]1)CCCC2)OC)OC C1(N(C)C(c2cnc(Cl)s2)=O)CN(C(C2(C)CCNC2=O)=O)CC1(C)C CCC(CC)CCC(C)(c1nnnn1C1CCOC1)NC1CCN(C)CC1 N1(C(c2c(CC)nccn2)=O)CCN2CCc3ccccc3C2C1 C(=O)(C(C(C)(C)C)n1cc(Cc2ncc(C)[nH]2)nn1)NC(C1CC1)C1CC1 N1(CC(=O)NC(CNC(c2ccc(CO)cc2)=O)C2CC2)CCC(O)CC1 c1(CC(N2C(CNC(COCC)=O)C=CC2)=O)cccc(C#N)c1 c1(C(N2CC(C(C)NC(C3(COC)CC3(F)F)=O)C2)=O)ccc(C(F)F)c(F)c1 c1(C(=O)NC(C(CO)NC(c2ccc(C)nc2C)=O)C)cncc2nnn(C)c12 c1(C(N(CC(O)CNC(=O)CC(C)(C)C2CC2)C)=O)ccc2nn[nH]c2c1 c1(C(=O)NC(C)(C)CCNC(=O)CCC2CCCC(O)C2)cc2n(c1)CCCC2 C1(OCC)COCC1N=c1[nH]c(=NCC(=O)N(C)C)c2ccc(OC)cc2[nH]1 C(=O)(CCCCCCC(=O)N(C1CN(C(=O)CC(F)F)C1)C)OC.C1CO1 C1(NC(Cn2cc(CNC(c3c(CC)cnn3C)=O)nn2)=O)CCCCCC1O N1(C(CC=CC)=O)CCC(NC(c2ccnc(C)n2)=O)C1C1CC1 c1(C(=O)NCC2C(NC(C(C)CN3CCOCC3)=O)C2)c[nH]c2cnccc12 C=CCCC(C)(C)C(=O)NCCC(C)NC(C1CC12CCOC(C)C2)=O c1(C(=O)NCC(C)(C)NC(C(CC)NC(N)=O)=O)cnn2c1CC(C)CC2 c1(C(N2CC(C)C(CNC(c3cncc(C(F)F)c3)=O)C2)=O)c(C#N)cnn1C C12(NC(CN(CCC)C)=O)COC(CNC(=O)CN3CCN(C)CC3)(C1)C2 c1(C(N2C3CN(C(C(CC)O)=O)C(C3)C2)=O)cnc2onc(C3CC3)c2c1 n1(C(C)C)ncc2c(N(C)C)[nH]c(=NCc3nccc(N4CCOCC4)n3)nc12 N1(C(CNC(N)=O)=O)CC2CCCC2(NC(=O)CCCc2ccc(Br)s2)C1 CC(CC(C)NC(C1(CCF)CCC1)=O)NC(=O)CSc1cnn(C)c1 C1(C(=O)OCC)CC(CSc2ccc(OCC#N)cc2)(CO)CC1.CCO c1(C(C(=O)NC(CC)C)N(C)CC2CCCCO2)sccc1Br C1(NC(C2CCC(C(N)=O)CC2)=O)CN(C(=O)Nc2ccccc2Br)CCC1F N1(C(c2cccc(OC)c2)=O)CCC(O)(CNC(C2CC(F)(CO)C2)=O)CC1 c1(C(=O)NC(C2CCN(C(c3cccc(N)c3)=O)C2)C)ccc2ncccc2n1 c1(C(=O)NC2CCC(N(C(CC=C)=O)C)C2)ccc(C(F)(F)F)cc1C c1(C(=O)NCC(CC(C)C)NC(=O)CC2CCNC(=O)C2)cc(Cl)ncc1N CCC(C)(O)C(=O)NCC(CCNC(=O)CCCOCCC)OC Cc1c(C(N2CC3(C2)CN(C(C2CC(C)(C)CO2)=O)C3)=O)sc2cccc(F)c12 C(N=c1[nH]oc2c1CC(C)CC2)C1(F)CCC(C)CC1 N1(C(C(C)(C)n2cccn2)=O)CC2(CCCC2NCCc2cnc(S)nc2)C1 C#CCC(CC#C)C(=O)N1CCC(N(CCO)C(c2ccc(O)c(C)c2)=O)C1 c1(C(N2CCC3CN(C(c4cn[nH]c4)=O)CC3C2)=O)cccc(O)c1[N+](=O)[O-] C=CCCCC(C(=O)NCc1ccc(F)cc1)N1CC2C(C(=O)NC)C2C1 C1(NC(CCCn2c(C)ncc2)=O)CC2(CCCN(C(=O)CN=S(C)(C)=O)C2)C1 c1(C(N2CC3(CCCN(C(CCCC)=O)C3)C2)=O)ccc(C)c(S(N)(=O)=O)c1 C1(NC(C(CCC)OC)=O)CCS(=O)(=O)C12CN(C(=O)CSCC)C2 Cc1occ2c1CC1OCCN(C1)C2C(=O)NCSC.C(F)(F)(F)COC C1(CNC(COCC)=O)CN(C(=O)C(=O)NCC2CC2)C(C)(C)C1 C12(NC(CC3CC(OC)C3)=O)CCC(C1)N(C(=O)C(c1ccc(F)cc1)C)C2 CC1CN(C(=O)C(C)CC(C)(C)C)CC(C)N(C(=O)Cc2cc[nH]n2)C1 N1(C(C2(CC=C)CC2)=O)CC2COCC(C1)C2NC(c1cc2cccn2cn1)=O C1(COC(C2(CCl)CCCC2)=O)(CO)CC2(CCC2)C1 N1(C(C2C(C)CC(C)O2)=O)CC(C)CN(C(c2ccnc(F)c2)=O)CC1C c1(C(C(=O)N(CCCCNC(COC(CC)C)=O)C)=O)cc(Cl)cc(Cl)c1 c1(C(C(=O)N(CC(CNC(C(C)(CO)OC)=O)(C)C)C)C)cccc([N+](=O)[O-])c1 C1(CC(=O)NCC=CC)CN(C(c2cccc(C(C)(C)C)n2)=O)CCO1 C=C(CNC1CN(C(N)=O)C1)C1CCOCC1 c1(C(N2CCC(O)(CCNC(CCC(CC)C)=O)C2)=O)cc(N)c(F)c(F)c1Cl C1(CNC(c2n[nH]c(C)c2F)=O)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CC1O C1(O)(CNC(CCc2ccc(C)s2)=O)CC2CCC(C1)N2C(=O)C(F)OC(F)(F)F CS(=O)(CC1CCC(F)(F)CC1)=NC(=O)Cc1ccc[nH]1 N1(C(c2c(C)oc(CNC(=O)CC3CCSC3)n2)=O)CCC(C)(C)CC1 C1(C(=O)NC(C)(CNC(=O)CCc2ccc(O)nn2)C2CC2)CCOC(=O)CC1 c1(OC)c(O)cc(C(N2CCCC(NC(C3CCCCS3)=O)CC2)=O)cc1C#N N1(C(Cn2ccc(C)n2)=O)CCC(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1C1CC1 c1(C(=O)CC2C(C(=O)NC3(CC=C)CCC3)CCC2)ccccc1[N+](=O)[O-] Cc1cc(C(=O)N(C2CN(C(c3cccc[n+]3[O-])=O)CCC2C)C)cc(C)c1Cl C1(C(N(CC(COC)(F)F)C)=O)CC(N=[N+]=[N-])CN1C(=O)C(C(C)C)C1CCC1 c1(C(=O)NC2C3CN(C(=O)CCCCC4CC4)CC23)ccnc2ccccc12 C1(CCC)CN(C(C2(C)CC2C)=O)CC1C(=O)NCCN1CCC(OC)C1 c1(NCc2c(C)nsc2)[nH]c(=NCCC(=O)NC2CCCC2)nc2scnc12 C(=O)(C(C)(C)CC(C)(C)C)N1CC(C(C)C)N(C(C2CN(C)CCO2)=O)CC1 n1(CC(=O)N(C2CCCCN(C(C=C(C)C)=O)C2)C)ccc2ccc(F)cc12 N#CC1CCC(C(N2CCOCC(C(N3CCCC3CC3CCC3)=O)C2)=O)CC1 C1(C(=O)NCC(CC)NC(C2(CO)CCCO2)=O)CC(C2CC2)=NO1 c1(C(C)=O)ccc(C(=O)NC(C)CNC(=O)CC2CCC3CC23)o1 C1(NC(CCSC)=O)CC(F)CN(C(=O)C(N)=O)C1 C1(NC(COC2(C#C)COC2)=O)CCC(NC(C2(C3CC3)CCCO2)=O)CC1 C=CC(CC)C(=O)NCC1(O)CN(C(=O)C(C)CC)C1 Cc1cnccc1OCc1cn(C2CCN(C(=O)C(C)(C)F)CC2)nn1 C1(C(C(=O)NC2C(NC(CCCOCC=C)=O)CCC2)F)CCC(=O)CC1 c1(C(N2CC(CCNC(=O)CN3CC4CC4C3)(OC)C2)=O)cc(Cl)cn1C(C)C C1(C(N2CCC(F)(CNC(C3NC(=O)OC3)=O)C2)=O)CC2CCC1CC2 C1(N(C)C(C23CC(CN2C(=O)CCCN=[N+]=[N-])C3)=O)CS(=O)(=O)C1(C)C c1(N(CCCNC(C2CCCCC2S(C)(=O)=O)=O)CC)ncnc2c1CCCC2 N1(C(CCC#CC)=O)C(C)CC2CN(C(C3CN(C4COC4)C3)=O)CC12 CCC(CC(=O)NC1CN(C(=O)CCP(C)(C)=O)CC1CC(C)(C)C)C(C)(C)C C(c1cncs1)=CC(=O)NC1CC(O)(CC)C1.c1(C(=O)NC2CCOC2)csc(C=O)n1 N1(C(C2C(NCc3c(C)scn3)CCC2)=O)CC(=O)N(C)C1 C(CCCCNC(=O)CN(S(N)(=O)=O)C(C)C)NC(c1csnc1Cl)=O c1(C(=O)NCC(C2CCOC2)NC(C(C)=CC)=O)cn(CCC)nn1 O(NC(=O)C=CCNC(=O)Cn1nccn1)CCC(C)O C1(OC)C(NC(=O)CC2C3CCCC3N2C(C2CCCCC2O)=O)CC12CCC2 C1(C(C)NC(=O)NC(C)(C)C)CCCN(CCCCN(C)C)C1 C12(CNC(C(CSC)C)=O)CCC(CC1)N(C(c1cnc3sccn13)=O)C2 CC(C(=O)NC(C)(C)CF)N(C(C1CCSC1)=O)C1CC1 c1(CC(=O)NC2CCCN(Cc3c(C)noc3C)C2)ccc(F)cc1Cl C1(C(N2CC3CC2C3C(=O)NCC(N)=O)=O)(CC)CCCCO1 C1(NC(c2n[nH]cc2C2CCC2)=O)CCCN(C(C2(Br)CC2(F)F)=O)C1 N1(C(C2(CCC)CC2)=O)CCOCC(C(=O)NC(C23CCC(CC2)C3)C)C1 N1(C(C(CCC)C)=O)CC(C)CCC1CNC(c1ccc(C(=O)NC)cc1)=O c1(NC(C2(c3ccc(C4CCC(=O)N4)cc3)CC2)=O)ccc([N+](=O)[O-])cn1 N1(C(C(CC#C)C2CC2)=O)CCc2cc(Cl)c(Cl)cc2C1C CC(C)C(C(=O)N1CCN(C(=O)C(C(C)C)n2cccc2)CC1)n1cccc1 c1(NC(=O)NCCC2(O)CCOCC2)ccc(O)c(=O)cc1 C12(C(N(C3CN(C(=O)CC4(O)CCCCC4)C3)C)=O)CC1Cc1c[nH]nc12 C#CC1CCCC(NC(=O)CNC(=O)CNC(c2cc(N)ccc2C)=O)C1 Cc1n[nH]c(C)c1CC(=O)NCCC1CCCCC1C(=O)NOCC1(C)CC1 Cc1cc(C=CC(N2CC(C)CC2C(=O)N(C)C)=O)on1.C1(CO)C(=O)N1 O=C(CCC(=O)NC1CC(NC(=O)CC2CCCCC2F)C1)c1ccccc1 c1(C(N2C(CNC(c3cccc(OC)c3F)=O)C=CC2)=O)ccc(O)c(F)c1F C(=O)(C1CC(C)(C)Oc2ccccc21)N1CC(NC(C(CC)CC)=O)(CO)C1 Cc1cc(C(C)C(=O)NCC2CC2NC(=O)CCCc2cc(C)no2)cc(F)c1 CCC(CC)C(=O)NC1CCC(N(C)C(c2ccc(OC(C)(C)C)nc2)=O)CC1 C1(C2CCN(C(c3csc(C4CCCO4)n3)=O)C2)(NC(c2cocn2)=O)CC1 c1(C(=O)NC2CN(CC(=O)NC)C(=O)C2)cc(C)c(F)cc1N N1(C(C2=NOC(C)C2)=O)CCC(C)(C)C(NC(C2CCC(C(F)(F)F)CC2)=O)C1 CC(CC(F)(F)F)C(=O)NC(C1CCCN1C(c1ccn(CCO)c(=O)c1)=O)C CC(C)C(CN=c1cc[nH]cc1S(=O)(=O)NCC(C)OCCOC(F)F)OCCO c1(C(=O)NC2(CCNC(C3C(C)C3C)=O)CCC2)cccc2ccoc12 C1(NC(=O)Nc2ccc(Oc3ccccc3)o2)CC(O)(CNC(=O)C(F)F)C1 N1(C(COC)=O)CCCCC12CC(NC(=O)CCNc1ccccn1)C2 CCC(C(=O)NC1(C(N2CCC(CC3CC3)C2)=O)CC(O)C1)SC C1(C(=O)NC(C=C)C(=O)OC)CCCC(OC)C1.C12(CC1)C(=O)N2 CN1CC2(CN(C(C3C4CC4CN3C(=O)CC3CC3(C)C)=O)C2)C1 Cn1nc(Cl)c(C(=O)NC(C(C)(C)C)c2ccco2)c1Cl C1(C(N2CCOC3(CC3)C2)=O)CC2CCC(C1)N2C(C1(Cl)CCC1)=O CC1CC(NC(c2cnc(O)o2)=O)CN(C(c2scnc2C(C)(C)C)=O)C1 C1(NC(C(C)N(C(CC2C(CC)C2)=O)C)=O)CC2(CCCO2)C1 Cc1cc(Cl)c(NC(Cn2cc(COC(c3cnn(C)c3C(F)F)=O)nn2)=O)s1 c1(C(=O)NCCn2ccc(C(=O)NCC(C#C)OC)c2)cccc(C(C)C)n1 c1(CC)c(C(=O)NC(C2(O)CN(C(c3cc(C)sn3)=O)C2)C)cnn1C CC(C)(CCNC(c1ccc(-c2cccs2)o1)=O)NC(C1CC1CF)=O C(=O)(C(C)C(=O)NC1CCCCC1C(N1CCCC1COC)=O)OC CC1CC(NC(c2cnn(C)c2)=O)CN(C(C2CCCCC2(C)C)=O)C1 N1(C(C=NOC)=O)CCOC2CN(C(c3nnc4ccccn34)=O)CC12 C(CCCC(C)(C)NC(=O)Cc1ccco1)NC(COCC)=O Cc1ccc(CC(=O)NC(C)(CNC(c2cncs2)=O)C2CC2)cn1 c1(N(CC(C)O)C)cc(S(=O)(=O)NC(c2ccccn2)CO)ccc1C#N CCCCC(C(=O)N(C)CCNC(=O)CC1CCC(C)(C)CC1)NC(N)=O C1(C(=O)NC2CN(C(CCS(C)=O)=O)CC3(C2)CC3)CC2CCCC(C1)C2=O c1(OCC(=O)NCCC2N(C(CCC=C)=O)CCOC2)cc(Cl)ccc1Cl C1(NC(c2nc(N(C(C(C)C)=O)C)sc2)=O)CN(C(=O)CN(C)S(N)(=O)=O)CC1F c1(C(=O)NC(CC)CN(C)C(c2cscn2)=O)ccnc(N2CCCC2)n1 S(=O)(=O)(c1cnc(NCC(c2ccccc2)CO)c(Cl)c1)NC(CCC)C1CC1 N1(C(c2c(CC)nccn2)=O)CC(CNC(=O)C(C)(C)COC(C)C)CC1(C)C c1(C(N2C(CNC(=O)CCCCO)CCCC2)=O)ccc2ccsc2c1 c1(CC)cnc(C(=O)NCc2nc(C(=O)NCC(C)(C)CN(C)C)c(C)o2)nc1 CC1CN(C(=O)CN(C(c2ccccc2F)=O)C2CC2)CC1n1cc(C2CC2)nn1 CN(CC1CCC1)N1CCCC(c2ccc([N+](=O)[O-])cc2)C1 C(CC(C)(C)C(=O)NCC1C(CO)C1(F)F)NC(c1c(C)coc1)=O C1(c2nnnn2C2CCCCC2)(NC2(CO)C(C)C2)CCCN2CCCCC12 c1(-c2cn(CC(=O)N(CC3CC3)CC3CC3)nn2)cccc(OC(F)(F)F)c1 CC1OC2(C(=O)NCC3CCN3C(=O)CCn3cnnn3)CCC1CC2 c1(OC)ccc(CN2CCOCC2C(F)F)cc1Cl c1(C(C(=O)NC(C)CC)N(C2CC(=C)C2)C)cc2cc(Br)cc(F)c2o1 c1(CC)ccc(C(N2CC(CNC(c3cc(C(N)=O)c[nH]3)=O)C(C)C2)=O)cn1 N1(C(=O)NC2(C)CCC2)CCCCC1CC1C2CN(CC(F)(F)F)CC12 c1(C(N2CCC(N(C(=O)C(C)C3CC3)CC#C)CC2)=O)ccc(C(C)C)c(O)c1 C1(NC(CCNS(CC)(=O)=O)=O)CN(C(c2occ3c2CCC3)=O)C2(CCC2)C1 c1(NC(C2CCC(NC(c3c(F)cccc3I)=O)CC2)=O)cnc2[nH]ncc2c1 Cc1[nH]nc2ncc(C(=O)NCC#CCNC(C3CCC(=O)O3)=O)cc12 C1(N(C)C(c2ccc(=N)[nH]c2)=O)CCC(NC(=O)CCC2CCCCCC2)CC1 C1(CNC(C(CO)NC(N)=O)=O)CC2CN(C(C34CCCC3C4)=O)CC12 C1(C(=O)NCc2ccc(CC)o2)(NCCC(=O)NCCCO)CCCC1C c1(C(N2CC(C)(C(=O)NCCC=CCCC)C2)=O)c[nH]c(=O)cn1 Cc1[nH]c2ccc(C(=O)NCC3CCCCN3C(c3sccc3F)=O)cc2c1C C1(C)(C(=O)NCCN(C(c2coc(C(C)OC)n2)=O)CC)CCC(=O)N1 c1(C(N2C(CN(C(C(C)(C3CC3)OC)=O)C)CCC2)=O)ccc(F)c2[nH]ccc12 N1(C(=O)OCC)CCC(C)N(C(C2CCC23CCCCC3)=O)CC1 C1(=C(C(=O)N(CCC(=O)NC2CCCC2)CC)F)CCCCC1 C1(C(=O)NC(C2(O)CCN(C3CCNC3=O)CC2)C)CCCCN1N=O c1(CNC(C(C)=CCC)=O)ccc(C(=O)N(C2CC2)Cc2[nH]nnc2C)o1 c1(N(CCC(F)CN)Cc2cc(OC)cc(OC)c2)c(C)cc(C)cc1C C(=O)(C(C)CCOCC)NC(C1(CC(=O)NCC2(OC)CCC2)CC1)C N(C(=NCCN1CC=CCC1)N1CCC2(CCCC2)CC1)C(CC)CC C1(NC(C2CCCC(OC)C2)=O)CCCN(C(=O)C(F)(F)C2CC2)C1C C#CCC(CC(F)F)NC(C1CCOCC1NC(C1CCC=CCC1)=O)=O c1(C(N2CC(c3ccccc3)(NC(=O)C(O)C(F)F)C2)=O)nnc(O)nc1O C1(Cl)(CC2CC(NC(=O)CSn3cc(-c4cnccn4)nn3)C2)CC12CCC2 N1(C(C(C)(C)c2cccs2)=O)CC2CCCC2(NC(=O)CC2CCCOC2)C1 c1(C(C(=O)NC(CN(C(C(C)NC(CC)=O)=O)C)C)(C)C)cc(Cl)ccc1F C1(C2CCN(c3nc(C)nc4sccc34)CC2)(NC(c2cnn(CC)n2)=O)CC1 C1(NC(c2cc3ccccc3nc2O)=O)CCCC2(CCCCC2)C1 CCC(CC(C)C)C(=O)NCC(C)=CC(=O)N(C)Cc1cnc(C)s1 c1(CC(=O)NC2C(CNC(CN(C3CCC3)C)=O)CCC2)ncn2c1COCC2 CC(CCNC(=O)COCC(=O)NC1(CF)CCC1)CCO CC1CCN(C(C2OCCCO2)=O)C(C)C1NC(C1CCC(C(N)=O)CC1)=O Nc1c(F)ccc(Cl)c1C(=O)NCC(CO)NC(C1(C(F)F)CCCC1)=O N1(C(C2(N(C)C)CC2)=O)CCC(F)(F)C(CNC(C2(C3CC3)CC=CC2)=O)C1 C1(CC)(NC(C2CCS(=O)(=O)N2)=O)CCCN(C(c2c(C)nc(C)n2O)=O)C1 N1(C(=O)CC2CCN(Cc3cc(O)ccc3Cl)C2)CCNC2(CC2)C1 c1(C(=O)NC2C(CNC(CCCOCC)=O)C2)ccc(Cl)c(C)c1N C12(NC(c3nn(C)c(Br)c3)=O)CCN(C(=O)CCC3CC(F)(F)C3)CC1C2 C(C(=O)NC1(C)CC(NC(C2CC2c2cccc(Cl)c2)=O)C1)(C(C)C)OCC C=CCC(CNC(=O)C(C)(C)CCSC)C(=O)N1CCCC(C)C1CC N1(Cc2c(C)noc2C)CC2CN(CC(N3CCC(C#N)CC3)=O)CC12 N1(C(=O)CCC2CCCO2)CCC(C(N2CCC(O)(CO)C2)=O)(CF)C1 c1(C(C)(C)C)ccccc1NC(C1CC1NC(c1ccc(F)nc1)=O)=O N1(C(C2CC(C(C)C)C2)=O)CC2(CNC(=O)CCC(N)=O)CC1(COC)C2 C1(NC(C2(OC)CCSC2)=O)CCCCC1C(=O)NC(c1ccccn1)CO C1(C(=O)NC(CN(C(=O)CN2C(=O)CCC2=O)C)(C)C)CN(S(=O)(=O)N(C)C)C1 CCN(OC)C(=O)CNC(=O)CC1CCCCN(C(=O)Cc2c(C)n[nH]c2C)C1 c1(C(N2CC(NC(CN(C3CCSC3)C)=O)C(F)C2)=O)cc2c(F)cccc2[nH]1 CC1CN(C(=O)C(O)Cc2cnc[nH]2)CC1NC(C1CC(N(C)C)C1)=O C1(C)(CC)CC(NC(C2CC(O)C2)=O)CN1C(c1cc(Cl)cnn1)=O C1(C(=O)OC)CN(N(C)C(C)c2cccnc2O)CC12CCOCC2 C1(C(=O)NC(COCC)C)CC2(CCN(C(C34CCC(C3)OC4C)=O)C2)C1 C1(NC(CN2CC(C)(C)C2)=O)CCN(C(=O)CC2CC(=O)NC2=O)C1(C)C c1(CCC(=O)NC2CC(n3cc(C(COC)(C)O)nn3)C2)ccc(O)nc1 C1(C(=O)NC2CC2)(CN)CCOC1.CC1CCCC(=O)N1C N1(C(CCNC(COC)=O)=O)CCCCCCC1C(N1C2CCCC1COC2)=O c1(OC)nc(NC2C3CN(C(c4ccc(Br)c(Cl)n4)=O)CC23)ncc1C N(C1c2ccccc2CC1NC(=O)CSC(F)F)C(C1C(C=C)OCCC1)=O C(=O)(C(C(=O)NCC(C)(O)CNC(=O)Cc1cccnc1)C1CC1)OCC N1(C(CC(COC)C)=O)CC(C2CN(C(C3CCC3c3nc[nH]n3)=O)C2)C1 CCC(C)C(C(=O)NCC1(C)CCCCC1O)NC(=O)CC(=O)NCC C1(C(N2CCC(N(C(=O)CNC=O)CC)C2)=O)CCc2cncn2C1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCC(C2(NC(=O)CC(C)C(F)F)CC2)C1 N1(C(C(C)NCc2ccco2)=O)CCCCC1CF c1(C(=O)NCc2scc(C(C)(C)C)n2)ccc2c(c1)CC(C)(C)O2 N1(C(c2ccsn2)=O)CCCC(C2CCCCN2C(=O)Cc2ccc(Cl)nc2)C1 C(=O)(C(O)P(C)(C)=O)NCc1cc(N2CCN(C(C(CC)OC)=O)CC2)ncc1 C12(CC)CCN(CC1)C(=O)c1c(cccc1)CNC2=O.C1(CO)CC2CCC1C2 C12(CNC(=O)Cn3nc(Br)c(Br)n3)CC(C1)C(C(=O)OC(C)(C)C)CO2 c1(C(=O)NC(CNC(COCc2nnc(C)s2)=O)C)ccc2c(c1)CN(C)CC2 N1(C(N)=O)CCCC(C(=O)NC2CN(Cc3cccc(O)c3)C2)C1.C(CO)O c1(C(=O)NC(CN(C(C(c2c(C)cccc2)C)=O)C)(C)C)ccn2c1CCCC2 C(=O)(C(F)CC(C)(C)C)N(C1(C(N2CCC(c3nn[nH]n3)C2)=O)CC1)C CC(C)CCC(C)S(=O)(=O)N1CCN(C2(C)CCC2)CC1 CC1CC(CC(=O)NC2(c3ccccn3)CC2)CN1C(c1ncccn1)=O CC(C)C(CNC(=O)CCC(C)n1ccnc1)C(=O)Nc1cccc2c1OCC2 S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CC(CNC(c2cc(F)c(F)cc2F)=O)C1 C1(NC(C(CC)OC)=O)CCN(C(C2CCC(=O)N2CC)=O)C1C N1(C(C2(OC)CC2)=O)CCCC(C2CC2NC(c2csc(CO)n2)=O)C1 CN1CCC(C)(C(=O)NC2CN(C(=O)Cc3cc(C4CC4)no3)CCC2F)C1=O C1(NC(CC2C=NN(C)C2=O)=O)C2CCC(C2)C1C(=O)NC(c1nc[nH]n1)C1CC1 C1(NC(C(COC)OC)=O)CCC2(CC1)CCN(C(C1(C(C)C)COC1)=O)C2 c1(N2CC(C)(CC)OCC2)nc(=N)[nH]c(=NCC2CSCCN2C(C)=O)[nH]1 C12(CNC(C(CCC)(C)O)=O)CCCC(CN1C(=O)CCSCCCCOC)C2 c1(C(N(CC(C)N(C(c2c(CC)onc2C)=O)C)C)=O)cc(C2CC2)cc(F)c1 CC1=C(C(=O)NC(CNC(=O)CSCc2cccnc2)C2CC2)CCCO1 c1(CC)ccc(C(=O)NC(C)CC(=O)NCCCc2nc(C)no2)cn1 C1(C2N(C(Cn3ncc(C)c3)=O)CCC2)CCN(C(C2CCC(C)O2)=O)CC1 C(CO)(C(C)NC(=O)CCSC(F)(F)F)NC(CCOCCC)=O C(=O)(C(C)CCC(C)(C)C)NC1CC(CC(=O)NCC(C(C)O)O)C1(C)C CCN(OC)C(=O)CNC(C1COC(CN)C1)=O.c1(C=O)ccc(=N)[nH]n1 CC1(C)CCC(CNC(c2cnc(C3CC3)s2)=O)N(C(C2CCCN2N=O)=O)C1 C(C(=O)NCC1(CC(=O)N(C)CC2CCOC2)CC1)(C(C)C)SCC C1(O)(CNC(=O)CC2(O)CCOC2)CCN(C(=O)C2=CCOC2)CC1 c1(C(=O)NC2CC(C)(NC(C=Cc3c(C)cccn3)=O)C2)nsc2ccccc12 C1(C(N(CC(=O)N(CCO)CCO)CC#C)=O)CCC(O)CN1C C(=O)(CC(CC)CC(F)(F)F)NCC(CC=C)NC(c1cc(C)n(C)c(=O)c1)=O C1(C(=O)N(C)CCc2cccs2)(NC(COCCC#C)=O)CCN(C)C1 N1(C(C(C2(O)CN(C(CCOCC)=O)C2)F)=O)CCC(N(C)C)C(C)C1 C1(NC(C2(CNC(C(C(=O)OCC)F)=O)CC2)=O)CCCC2(CN(C(C)=O)C2)O1 N(C1CCCc2cccnc21)(C(=O)C(=O)NCCC(F)(F)F)CCC Cn1cc(NC(=O)C(c2ccccc2)=O)cc1C(=O)Nc1cncs1 C1(CNC(C2C(C)=CCS2)=O)(NC(=O)CCOCC(F)F)CCCCC1C c1(NC(C)CCNC(c2ccc(C(=O)OCC#N)cc2)=O)ncccc1[N+](=O)[O-] C(=O)(CC(C)CC(=O)NCCC1CCCCN1C(c1cncn1C)=O)OC C1(CC)CN(C(c2cnc(Cl)[nH]2)=O)CCC1NC(c1cnc(C(C)C)[nH]1)=O c1(OC)ccc(C(N2CCCC(N(C(=O)C#CC3CC3)CCO)C2)=O)c2ccncc12 C1(NC(C(CC)=CCCC)=O)CC2CCC(C1)N2C(C1CCO1)=O C1(C(=O)NC(c2cnn(C)c2)C(=O)N(CC)Cc2cccs2)CC2C=CC1C2 Cc1ccc(N(C(=O)C(C)CC(=O)O)C2CCOC(C)C2)c(C)c1 C(=O)(C1=C(C)OCCS1)OC.C12CCC(C1)N(CCS(N)(=O)=O)C2=O Cc1nc(C(=O)NC23CCN(C(=O)CCc4cnn(C)c4)CC2C3)c(=O)[nH]c1C C1(OC)CCN(C(c2ccn3ccccc23)=O)CC(C)(C)C1 C1(C)(CC(=O)NCc2ccc(C(N(CC(F)CO)C)=O)s2)CCOCC1 C1(CCNC(=O)C(O)Cc2ccccn2)(OC)CN(C(=O)C(C)c2cc[nH]n2)C1 CC1(NC(CN2C(C(=O)NCc3ccccc3)CCCC2)=O)CS(=O)(=O)C1 C1(C(=O)NCCC(C)NC(c2c[nH]c(C#N)c2)=O)CNC(=O)N1C c1(C(N2CC(C)C(CCNC(=O)C(F)=C3CCC3)C2)=O)cnn2cccc(Cl)c12 C1(C(N(C)CC)=O)CCCN(S(=O)(=O)CC)C1.N12CCCC1SC(C)C2=O c1(NC(C(C)OCCCC)=O)cc(C2CC2)nn1C.C12CCC(C1)CNC2=O C1(C(=O)NC)CCN(C(=O)CC2CC(OC)C2)CC1 c1(C(C(C)Sc2nnc(C3CCC3)n2C2CC2)=O)cc(Cl)cc(Cl)c1 N1(C(c2cc(NC(C)C)ncc2)=O)C2CCC1C(CNC(c1cocn1)=O)C2 Cc1ccnc(CNC(=O)CCN(C(c2n[nH]c(C)c2Cl)=O)CC2CC2)c1 C1(NC(c2ccc(C3CCCO3)[nH]2)=O)CC2CN(C(C3C=C3C)=O)CC2C1 c1(OCC=C)ccc(Cl)c(CN2CC(O)CC2C(N2CCCC(F)(F)C2)=O)n1 C1(NC(C2(C)ON=C(C)C2)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)cc1)C2 C1(CNC(C(n2ccc(C(F)(F)F)n2)C)=O)CCCCN1C(=O)COCC(F)F Cc1[nH]c(=NCCCCC(C)NC(=O)C(C)Cc2ccc(Cl)cc2)ccc1C#N c1(CN(C(c2cccc(Cl)c2)CCO)C)ccc(C(C)(C)C)cc1 C#Cc1cccc(C(=O)N(CC(C)N(C(=O)CN2C(=O)CNC2=O)C)C)c1 c1(CC(=O)NCC2(O)CC(NC(CC(C)C)=O)C2)cn2ccccc2n1 N1(CCCC)C(=O)CC(NC(=O)NC(c2nc(C(F)(F)F)c(Cl)s2)C)C1=O C1(C(N(C)CCn2cncn2)=O)CCC2(CC2)N1C(c1ccc(C#N)n1C)=O C#CCC(C(=O)N1CCC1(C)CC(=O)NC(C)CN1CCCC1C)C1CC1 N1(C(C=CCN(C)CC)=O)CC(CC(=O)NC2COC(C)(C)C2)C(C)C1 c1(N(C)C)ncccc1C(=O)N(C1CCN(C(C2CNC(=O)C2)=O)C1)C N1(C(c2ccc(C#C)cn2)=O)C2CCC1CN(C(c1nccn1C(C)C)=O)C2 Cc1cocc1C(N1CC=CC1CNC(c1cncn1C)=O)=O c1(C(=O)NCC(CC)(CC)NC(=O)Cc2[nH]cnc2C)ccc(C(C)C)nc1C CC1CC(C(=O)NCCCCC(=O)N2CCS(=O)CC2)CC(=O)N1 C1(CNC(CCCC=C)=O)CCN(C(=O)C(=C2CCCCC2)F)CC1C c1(C(=O)NC2CC(N(C(c3c(CC)n(C)nn3)=O)C)C2)nc(O)nc(O)c1N C#CCC(C(N)=O)NC(C1C(CC(=O)NC)C1)=O.C(=O)(CCC)N C(C(F)(C(=O)N(CC(Cl)Cl)C)C(C)C)NC(c1c(CC)ncnc1)=O CC1=C(C(=O)N2CCN(C(=O)CN(C(=O)CC3C(=O)ON=C3C)C)CC2)CCC1 c1(CC)nnc2cc(N3CCCC(NC(=O)CCc4nc(O)n[nH]4)C3C)ncn12 c1(C(C)=O)ccc(S(=O)(=O)N2CC(C)(CNC(c3cc(O)n[nH]3)=O)C2)cc1 c1(C(=O)Nc2ccc(NCCn3cc(Br)ccc3=O)cc2)cccc2c[nH]nc12 N1(c2nc(C)nc(=N)[nH]2)CCCC2(NC(C3CCS(=O)(=O)N3)=O)CC2C1 c1(C(=O)NCC(CNC(C(OC)OC)=O)CO)ccnc(-n2cccn2)c1 c1(OC)nc(C)cnc1C(N1CCC(CO)(CNC(C2CCCCS2)=O)CC1)=O N(C(=NCC1CCC1)NC(C1CCCCC1)C1CCCO1)CC1N(CC)CCC1 N1(C(CC2CC(SCC)C2)=O)CCN(n2cc(C3CCN(C)C3)nn2)CC1 C12CN(CC3CCCC13)C2=O.C1(C(=O)NC(=O)C(F)(F)F)CN=C2N=CNN2C1 c12nc(=NC3CC3C)c(c[nH]1)OC(=O)C2.CC C1(NC(C(F)OC)=O)CN(C(=O)C2=CCSC2)CC1F N1(C(C(CSC)C)=O)CC2(CC(NC(c3cnsc3C)=O)C2)C1 c1(C(=O)NC(CNC(C(C)N2CCC2)=O)(C)C2CCC2)ccn(C)c1 c1(NC(C2CC2CNC(C2COCCO2)=O)=O)ccc(-c2ccccc2)nn1 N1(C(c2ccc(C(F)(F)F)s2)C(=O)NCCCC)CC(C(F)(F)F)CC1C CC(C)C(C#N)C(=O)N(C)CC1C2CN(C(=O)COCC3CCCO3)CC12 Cc1nn(C)c2c(NCC3(CCCO)CC3)nc(N3CCOC(C)(C)C3)nc12 c1(C(N2C(CNC(C3N(CC)CCC3)=O)CC2)=O)cnn2c1CCCC2 c1(CC)ccccc1S(=O)(=O)N1CCCC1CNc1ccc(Br)c(C)n1 CC1(NC(c2nnc(C3CC3)s2)=O)CCCN(C(C2(F)CCCCCC2)=O)C1 N1(C(CC2C(CC)C2)=O)CC2(CC(NC(c3ccccc3Cl)=O)CO2)C1 C1(NC(CCSCC(=O)OC)=O)CCCC2CN(C(C3CCCC34CCC4)=O)CC12 C(=O)(CCCCC#N)NCc1c(C(N2C(C(C)C)CC(O)C2)=O)cco1 c1(C(C(=O)N2CC(CNC(COCCC=C)=O)C2)C)ccc(SC(F)(F)F)cc1 CCCC(C(O)C(=O)N(C1CCN(CC)C1)C)NC(C1CCSCC1)=O c1(SCC(=O)NC(CC=C)CNC(c2cn(CCC)nn2)=O)ccccc1C c1(CNC(=O)Nc2ccc(CC)nc2)cc(C)c(F)c(C)c1 C1(NC(C2CCOCC2)=O)CN(C(=O)CN2CCSCC2)CC1n1ccnn1 C1(CCCC)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CCN1C(c1coc(Br)n1)=O c1(C(N2CCC(C)N(C(=O)CC3(C)CCCC3)CC2)=O)ccc2c(c1)COCC2 C1(NC(CCSC)=O)CCN(C(=O)CN2CCOCC2)C1C1CC1 C=C(C)C(C)(C)C(=O)NCC1(O)CC(NC(c2cc(Cl)ccn2)=O)C1 C1(CN(C(C2(C(C)NC(C(C3CCC3)OCC)=O)CC2)=O)C)COC(C)(C)C1 CN1CCN(C(c2nocc2Cl)=O)CC1C(=O)NC(C1CCC1)C1CC1 C1(NC(C(C)NC(CC)=O)=O)CCCCCN(C(=O)CC2CCCCCC2)C1 c1(OC)ccc(CC(=O)NC(C)C(c2ccc(Cl)cc2)O)cc1[N+](=O)[O-] N1(C(c2ccc(OC)nc2Cl)=O)CCC(C2CC(NC(=O)CC(C)C)C2)C1 c1(C(=O)NCC(CN(C(Cn2c(C)nnn2)=O)C)O)cc(C(F)(F)F)ccc1Cl CCCC(CC)N=c1cc(C)[nH]c(=NCC(C(C)(C)C)c2ccccc2)[nH]1 Cc1nc2cc(C(N3CC4CC(NC(c5ccncc5C)=O)C4C3)=O)ccc2s1 C1(C(=O)O)CN(C(=O)CO)CC1c1ccccc1.C1CCOCC1 c1(C(=O)NCC2N(C(C(CC)(C)CC)=O)CC2)cnn2c1CCCC2C C1(C(c2nnnn2C2CC2)NCC(c2ccc(F)cc2)C)CCC2CC1C2(C)C c1(C(=O)NCCCN(C(=O)C=Cc2nccnc2C)CC)cc(C)cc(C#N)c1 O=C(NNc1ccc2c(=O)[nH]ccc2c1)C(F)(F)c1ccc(Cl)c(Cl)c1 N1(C(CCCCCN(C(C2=C(C)CCC2)=O)C)=O)CCCNC(=O)C1C(C)C Cc1ccc(Cl)c(NC(=O)C(=O)NC2CCCN(C(=O)CC3CCCNC3)C2)c1 c1(C(N2CC(C)C(C(=O)N(C3CCSC3)C)C2)=O)ccc(N)c(F)n1 Cc1cscc1C(=O)N(C)CCN(C(=O)CSCC(c1ccccc1)C)C C(=O)(CC(=O)NCC1CCC(NC(c2[nH]nnc2C)=O)C1)NCC#C c1(C(N2C3C(CC(=O)Nc4ccc(OCF)cc4)C(C3)C2)=O)ccc(Br)c(Cl)c1 C(C(=O)NC1CC1NC(c1cccc(O)c1C)=O)(C(C)(C)C)NC(C)=O C(C(C)CC(=O)NCCn1cc(C(N2CC=CC2CF)=O)cn1)OC c1(NC(CCCCC)c2nnnn2-c2ccccc2Cl)cc(Cl)cc(Br)c1 c1(C(N(CCC(C)CO)C)=O)ccc(OCc2ccccn2)nc1 C(CCCCC(=O)NC(C1CCOCC1)C)NC(CC(C)CN(C)C)=O Cc1ncnc(C(=O)NCC2(F)CCCN(C(C3(C#N)CC3)=O)C2)c1C C1(C(CNC(c2cc(COC)sc2)=O)C)CCN(C(=O)CC2(O)CCCC2)CC1 C1(O)(CNC(c2c(C)cco2)=O)CCCN(C(=O)Cn2ccccc2=O)CC1 C(c1ccc2c(c1)COCC2)=CC(=O)NCC1CN(C(CN2C(C)CCC2)=O)C1 C1(C(=O)NC2C(CC=C)COC2)CCC(C(C)C)N1C(=O)C(C)CN(C)C c1(OC)nc(Cl)ccc1C(=O)NC1CC(C)CN(C(=O)CCc2ccoc2)C1 C(C(C(C)(C)C)NC(=O)CC1(C)CCCCC1)NC(CN(C1CC1)CC)=O c1(CC)cccc2oc(N(C)C)nc12.c12ccc(cc1)C(C)(CC)NC2=O c1(C(N2CC3CN(C(c4c(C)nco4)=O)CC3C2)=O)cc2cc(Br)cnc2s1 c1(C(C)NC(=O)N(C)C)cccc(Br)c1Cl.c12ccc(cc1)C(=O)COC2=O C(C(C(=O)NC1C=CCCCC1)C(C)C)NC(C(CC)CC)=O.O1NS(=O)(=O)N1 C1(NC(C(C)(C)OCC)=O)CCOCC1C(=O)NC1CC(n2cccn2)C1 C(=O)(C1CCCn2ccnc21)N1CCC2CN(C(c3ccc(C)c(C)n3)=O)CC21 C1(CNC(CN2CC(C)(OC)C2)=O)(CNC(=O)CC2(C)CC2)CC2CCCC2C1 C1(C(N2C(c3onc(C)n3)CCC2)=O)CCCCN(C(C2CCCC(C)C2)=O)C1 C1(COC)(CNC(C2CCSCC2)=O)CCCN1C(C1CCC(C)O1)=O C(C)(CC(C)N=c1nc(C)nc2[nH][nH]cc1-2)NC(C(CCC)C)=O c1(SC)cc(C)ccc1C(N1CC(N(C(=O)CC(C)F)C)C2(CC2)C1)=O CC(Cc1cnc[nH]1)C(=O)N1CC(CC(C)NC(=O)CN(c2ccncc2)C)C1 N1(C(=O)Nc2cccc(C)c2Cl)CCCC2(CNC(=O)C2)C1 c1(NC(c2cc(C(F)(F)F)cc(F)c2)=O)ncc(Br)nc1Cl.C12CC1CNC2=O CC(O)C(F)(F)C(=O)NCCCOCCNC(=O)COCC1CCCOC1 C1(N(CCCCC)C(C2COC(C3CC3)C2)=O)CCN(C(=O)CCC)CC1 C1(S(C)(=O)=O)(C(=O)NCC2C(NC(c3ccc(C)c(F)c3N)=O)C2)CCOCC1 c1(CC)ccc(C(N2CC(O)(C(C)NC(=O)C(C)CCN(C)C)C2)=O)c(F)c1 c1(C(N2CCC(C)N(C(=O)COC3CCC3)CC2)=O)ccc2c(Cl)nccc2c1 Cc1c(Cl)ccnc1C(N1CCOCC(NC(c2nn[nH]c2Cl)=O)C1)=O C1(CNC(CN(C2CC2)CC)=O)CCCCN(C(C2CCN(CC(C)C)C2)=O)C1 C12(C(=O)NC(CNC(C(C)(C3CC3)OC)=O)C3CC3)CC3CC1C2C3 C(C(CC=C)C(=O)NCC1(F)CC(CO)C1)NC(C(CC#C)O)=O N1(C(CNC(c2c(OC)oc(-c3ccco3)n2)=O)=O)CCN(C(C)=O)CCC1C CN1CCC(C(N2CCC(CC(N3CC(OCC(F)F)C3)=O)CC2)=O)C1=O C1(NC(C2N(CCC)CCCC2)=O)CCN(C(=O)CC2CCCCC2)CC1F CCC(C)(CC)C(=O)NC1CC1NC(c1cccc(-c2ccncc2)n1)=O CC(C(=O)NNC(=O)COc1nc(NCNC(C)(C)C)c(F)cc1)c1ccccc1F C(=O)(CC1CCOc2ccccc21)NC1CCN(C(CC(C)CC(C)(C)C)=O)C1 c1(C(=O)OCC)cnn(-c2ccc(C)cc2)c1NC(=O)C(C)N(C)C(C)=O c1(OC)ccc(C(=O)NCC2(OC)CCN(c3ccncn3)CC2)c(OC)n1 O(NC(=O)CC(C)(C)C)C(C)C#N.C(=O)(CCN=[N+]=[N-])N c1(C(=O)NC(CC)CNC(=O)Cn2ncccc2=O)ccc2c(c1)OCCN2 C1(C(=O)N(C2CC(C(=O)NCC3(CO)CC(C)(C)C3)C2)C)(OC)CCCOC1 C1(N(C)C)CN(C(c2cccc(Cl)c2Cl)C#N)CC12CC2 CC(CN=c1cccc(S(=O)(=O)N2CCCC(OCCO)C2)[nH]1)C(C)(F)F C(C)(COC(C)=O)(CC(=O)O)NCc1cn(CCCC)nn1 NC(=O)CCC(=O)NCCC1CCCN1C(C1SCCCS1)=O C1(C(=O)NCCCCn2cc(C3CCOCC3)nn2)Cc2ccccc2NC1=O C1(C(N(CC(C)C)C(C)CO)=O)CC12CCCC2 C=CC(CC)CC(=O)N(C)CC1CCCN(C(=O)Cc2cc(C)ns2)C1 N1(C(c2ccc(CSC)o2)=O)CCC(NC(C2CC3CCC2O3)=O)C1C Cc1ccc(F)c2c1CCN(Cc1cn(CC3CCNCC3)nn1)C2 c1(NC(C2N(C(c3c(CC)occ3)=O)C3C(C2)C3)=O)cc(CC)ccc1O C1(NC(c2ncn(C)c2)=O)CCN(C(c2cc(C(F)(F)F)ncc2Cl)=O)CC1F CCCCC(C(=O)NC1CCC(F)(CNC(C2(S(N)(=O)=O)CCC2)=O)C1)C(C)C n1(-c2c(C)cccc2)cc(C#CCNC(=O)C(C)OC2CCCCO2)nn1 C1(CNC(=O)NCC(n2c(C)cc(C)n2)C)CC(C2CC2)=NO1 Cc1nn(C)cc1CCC(=O)N(C)CCOCCNC(=O)CC1CC1C c1(C(=O)NC2C=CCN(C(CCC3OCC(C)(C)C3)=O)C2)ccc2snnc2c1 c1(C(=O)NC2(Cc3ccccc3)CC23CCC3)cccc2c1OCO2 N1(C(c2n(CC)ncc2)=O)CCCC(C(=O)NCCCC(=O)OC)C1 C(=O)(CCCCCN=[N+]=[N-])NCCCCCCC(=O)NC1CC(C)OC1=O C=CCC(CCCCC)C(=O)NC(C#N)C(=O)O C1(NC(C(CC)(F)F)=O)CN(C(C2CC23CCOCC3)=O)CC2(CC2)C1 Cc1c(C(=O)NC2CCN(C(=O)C3CC3)CCC2CO)[nH]c2cc(F)cc(F)c12 CC1(C)Oc2ccsc2C(NC(=O)C(=O)NC(c2ccccc2F)C)C1O C12(NC(c3nccc(C)c3)=O)CCC(CNC(=O)CCCC(C)C)(C1)OC2 C1(C(N2CC[Si](C)(C)CC2)=O)CC2CCCC2N1C(=O)CN1CCCCC1 C1(CNC(c2cccc(CC)n2)=O)C(C2CC2)CCN1C(=O)C(F)OC Cc1nc(C)c(C(=O)NCC2(C)CCN(C(=O)CCc3ccccc3)C2)[nH]1 C12(CNC(c3c(CC)nccc3)=O)CC(CO1)N(C(C1CC(=O)NC1(C)C)=O)C2 c1(CC)ccccc1OCC(=O)NC1CCC(C)(NC(=O)C(C)COC)C1 C(C(C(=O)NC(CC1CCCC1)C(=O)O)N(C)C)NC(C)=O C(=O)(C1=CC2CCCC12)NC(C1CCCCN1C(C1CC2CC2C1)=O)C C1(C)(C(N2CCC(CC(N(C3CC(=C)C3)C)=O)C2)=O)CCCCC1 c1(C(=O)NCC(C)NC(c2c[nH]nc2C(F)(F)F)=O)scnc1Cl N1(C(C2CCCN(C(C)=O)C2)=O)CCN(C(c2ncn(C)n2)=O)CC1C1CC1 N(C1CCn2ccnc21)C(=O)Cc1ccc(OC2CC2)cc1 O=C(CCCC(F)F)N1CC(n2cc(-c3cccs3)nn2)C(O)C1.C1C(=O)N1 c1(C(N2CC(F)(CNC(c3cc(Cl)cc(Cl)c3)=O)C2)=O)ccnc2[nH]ncc12 c1(C(N(CC(C)NC(c2ccnc(C(F)(F)F)n2)=O)C)=O)ccc(Cl)cc1 N1(C(C2C(CNC(C(CSC)(C)C)=O)C2(C)C)=O)CC2CCC(CO)(C2)C1 Cc1ccc(C(=O)NCC2(C(C)NC(c3sccc3Cl)=O)CC2)o1 c1(C(N(C2CCN(C(C3(F)CCCC3)=O)C2)C)=O)ccc2nc(CO)[nH]c2c1 C1(C(N(CC(C)C)C)=O)CCC(C)N(C(=O)CCC2CCCCO2)C1 c1(C(=O)NCC2(NC(C(C)=C(CC)C)=O)CC2)nccc2nn[nH]c12 C(c1ccc(C(=O)NCC(F)CNC(C2(NC=O)CCC2)=O)cc1)=CC(=O)O c1(OC)cc(N2CCC(CNC(C3CC3F)=O)C2)ncn1 CC1CC(=O)NC1C(=O)NCC1CCC(C(=O)NC2C(C)CCC2C)CC1 C(=O)(CC1OCc2ccccc21)N1CC(O)(CNC(C23CCC(C)(OC2)C3)=O)C1 C1(C(N2CCn3c(CCO)nnc3C2)=O)CC12CCS(=O)(=O)CC2 c1(CCC(=O)NC(CNC(C=C(C)C(C)C)=O)C)cnc(O)[nH]1 N#Cc1cc(Br)cnc1N1CCC(Nc2ccc3occc3c2)C1 C1(NC(CCSCC)=O)CC12CCN(C(=O)CN1CC(C)C1)CC2 CC(C1CCCCC1)=CC(=O)NC1(C)CCN(C(C2CCC2C(C)(C)C)=O)CC1 N1(C(CCNS(CC)(=O)=O)=O)CC(F)(F)CC1CCNC(C1CCN1C)=O Cc1nc(CCNC(=O)COC2CN(C(=O)Cc3ncoc3C)C2)n[nH]1 C(=O)(C1=C(Cl)CCC1)N1CCC(N(C(c2cnn(C)c2Br)=O)CC)C1 c1(C(=O)NCCCNC(CC2C(C)(C)CCO2)=O)cccc(N=S(C)(C)=O)c1 N(C1CCCOc2c(Cl)cccc21)C(C(COCC)n1cc(CO)nn1)=O C=CCCC(=O)CN1CC(c2ccccc2C)C(O)C1 CCCCC(F)C(=O)NC1CCN(C(=O)CCn2cncn2)C(C)C1 CC1CCC(NC(C2(c3ccccc3)CC2)=O)CN1C(=O)CSCC1CCCO1 N1(C(C(C)CS(C)=O)=O)CCc2c(c(CNC(c3nnc(S)n3C)=O)nn2C)C1 C1(C(N2CC(N(C(C=Cc3cnc(C)s3)=O)C)C2)=O)C2(CC2)C12CC2 C(C(C)(C)C(=O)NCC1CN(C(=O)C(c2ccc(C(C)(C)C)cc2)(C)C)C1)OC CCC(CCCC(=O)NC(c1ccns1)C)NC(C1(OC)CCOC1)=O C1(NC(CC(CC)Cc2ccccc2)=O)CN(C(C2CCC2)=O)CC2(CC2)C1 Cc1cc(F)cc(Br)c1N(C(C)(C)C)CC(F)F.N12CCC(CC1)N(C)C(=O)O2 N1(C(=O)Nc2c(C(C)C)cccc2)CC(CO)C(F)(COCc2cccnc2)C1 C=CCN(CCN1CCOCC1)N1CCOCCOC(C2CC2)C1 c1(C(=O)N(O)Cc2cn(-c3cncc(Cl)c3)nn2)nc(Br)n2c1COCC2 N12CCCN(CC1)C(=O)C2=O.Cc1cnc(C(C)N(C2(C3CC3)CC2)C)s1 c1(C(N(CCC(C)NC(=O)C=CC2CCC2)C)=O)ccn2c1CCCC2 c1(C(CC)NC(=O)C(N2CCC(CO)C(O)C2)=O)cc(F)c(F)cc1OC N=c1nc(NC2CC(NC(C3CC=CCC3)=O)C2)[nH][nH]1 C1(C(=O)NCC(CN(C(c2c(CC)ocn2)=O)C)(C)C)COCCC1(F)F C1(NC(C2CC23CCN(C(=O)Cc2cncnc2O)C3)=O)CC2(CCOC2)C1 C1(O)(CN2CC(N(C(c3nnn(CC)c3C)=O)C)C2)CCCC(C)C1 C1(CNC(C(CCC)CC)=O)CN(C(C2(C(=O)N(C)C)CC2)=O)CCC12CCC2 c1(OCCC)ccc(COCCNC(=O)NCCS(=O)CC)cc1 C(C)(CC(C)(C)OC)NC(C(COC)Oc1ccc(Br)s1)=O C1(C)(NC(c2ccc(CNC(C(c3cnn(C)c3)C)=O)[nH]2)=O)CCC(O)CC1 N1(C(C(Cn2ccc(C)n2)C)=O)CCC2(C1)CN(C(C1(C)CCOC1)=O)CCO2 C(=O)(CCC(C)(C)NC(=O)C(C)(C)CF)NC(C1CCN(C(=O)C2CC2)CC1)C C(CC)(CCC(=O)NC1CC(N(C)C)C1)NC(CNC(CCC)=O)=O C1(NC(C2C(C)C2)=O)CCCC12CN(C(c1cnn3c1OCC3)=O)C2 N1(C(C(C=C)(C)CC)=O)CC2CCCC(NC(c3ncc(C(F)F)s3)=O)C2C1 C(=O)(CC(C(F)F)c1ccccc1)N(CCN(C(C(C)=CC)=O)C(C)C)C Cc1oc(C(=O)OC(C(N2CC(NC(=O)OC(C)(C)C)C2)=O)=O)nc1C1CC1.NC.OC N1(C(C)=O)CCN(CCC)CC1.c1(C(C)C)nc(CNC(=O)CC2(C)CC2)cs1 Cc1nn2cc(C(N3CCC(CO)(NC(c4ccc(C(N)=O)s4)=O)C3)=O)nc2s1 Cc1oc(Br)cc1C(=O)NC1CCN(C(c2nn(C)cc2Cl)=O)C1C1CC1 C1(C(=O)N(C)CCC2CCC2)(CC)CCN(C(C2CCCCC2C)=O)CC1 O=C(C1=CC(O)CCC1)N1CC2CCN(C(c3ncoc3CCC(F)(F)F)=O)C2C1 c1(N(c2cc(-c3cnn(C)c3)ncn2)CCC)cc(C)ccc1C(F)(F)F c1(C(N(CC(CC)NC(C)=O)CC)=O)cc(NC(=O)CC(F)(F)Cl)cnc1C N1(C(c2coc(Cl)n2)=O)CCC2C(CCCN2C(c2[nH]nc3ncccc23)=O)C1 C1(NC(COCc2cc(C)n(C)n2)=O)C2CCN(C(C3(CF)CC3)=O)CCC12 Cc1cc(NC(=O)CN2CCC(C(C)(C)O)C2)ccc1F S(=O)(=O)(c1cccc(Br)c1)N(C(c1cc(C)cc(C)c1)C(=O)O)C N1(C(c2ccc(C#C)s2)=O)CCC2(NC(=O)COc3ccc(F)nc3)CC2C1 N1(C(c2cc(C)nc(C)c2)=O)CC2(CNC(C3CCS(=O)(=O)C3)=O)CC(F)(C1)C2 NC(=O)CCCN(C(=O)C(N)CC1CC1)c1ccccc1 C1(CC(=O)NCC(C)CNC(c2cncc(Br)c2)=O)CCC2(CCC2)O1 C1(C(=O)NCCCn2cc(CCCCCCO)nn2)CCCCC12CC2(F)F c1(NC(=O)C(N2C3CC2CN(Cc2ncc[nH]2)C3)=O)ccn2ccnc2c1 Cc1cc(C(N2CCC2NC(C23CCC(CF)(CC2)CC3)=O)=O)c(Br)c(C)c1 C(=O)(C=C=C(C)C)N1CCC(CCC(=O)NCC(C(=O)OC)O)C1 C1(N(C(c2[nH]nnc2C)=O)CC)CCCN(C(=O)C(C)(C)n2ccc(C)n2)C1 C12(CNC(=O)C(F)C3CCC3)CC(CO1)N(C(=O)C=CSc1ccccc1)C2 c1(C(=O)NCC(CNC(CCCOCCOCC)=O)F)c(N)cc(Cl)cc1F c1(NC(c2cccc(OC(C)=O)c2)=O)cc(C)nc2ccnn12 N1(C(C2C(C)=CCS2)=O)CCCC(c2n[nH]c(CNC(=O)C(C)C#N)n2)C1 c1(C(=O)NC2CC3(C(NC(C(CC#C)O)=O)C3)C2)cc(C(=O)OC)cc([N+](=O)[O-])c1 C1(C(=O)NCC(CCNC(CNC(=O)OCC)=O)O)CCCCN1C c1(CC)nn[nH]c1C(=O)NCCNC(c1cc(C)[nH]n1)=O.c12cn(nn1)C2 CC1CCN(C(C2CCS(=O)(=O)CC2)=O)CC1NC(=O)C(c1cccc(F)c1)O N1(C(=O)NCc2ccc(CC(N3CCCC(C)C3)(C)C)cc2)CC2(CCC2O)C1 Cc1ccnc(C)c1C(=O)NCC(N1CCN(C(C2(CO)CCC2)=O)CC1)(C)C N1(C(C2CC(F)(CO)C2)=O)CCN(C(C2CCCCS2)=O)C(c2cccnc2)C1 CC1(C)CCCOC1CC(=O)NCC1CN(C(=O)CCC(F)F)CCC1CO C1(C)(COC)CC(NC(c2cccc(C)n2)=O)CN1C(c1cnco1)=O c1(C(=O)NC(C2CC(F)(F)C2)C)cccc(-n2cc(CC3CC(F)(F)C3)nn2)c1 C=C(C)CCCC(=O)N1CCC(CO)(CNC(=O)CCOC2CC2)C1 c1(C(=O)NCC2CN(C(COc3cccc(C)c3)=O)C2)cn2ncccc2n1 c1(C(N2CCC3(NC(=O)CCCCC4CC4)C(C2)C3)=O)ccc2nccn2n1 N1(C(CC)=O)CCN(C(=O)C(CCSC)NC(c2cn(CCO)nn2)=O)CC1 C1(C(=O)NCc2ccc3nc(C)sc3c2)CC(O)c2ccccc2O1 Cc1cc(CNC(C2(CF)CC2)=O)ncc1Br.C12CCN(C1)C2 N1(C(CCOCCC)=O)CCOCC(NC(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 c1(NCC(c2scc(C)n2)C)cc(N(C)CC2CCC2(F)F)nc(C(F)(F)F)n1 C12(C(N3CC(C(C)NC(=O)Cn4ncc(O)nc4=O)C3)=O)CCCN(CCC1)C2 C=C(Cl)CC(C(=O)N(CCCSC)C)NC(=O)CN1CCOCC1=O C1(C(N2CCC(CC)C2)=O)CCN(C(=O)C(C)N2CCCC2)CC1 C1(CCC(N2CCC(n3ccnc3)C2)=O)CCCCN1C(=O)Cn1cccc1 CC(C(=O)N1CCC(OCCOC2(CCN=[N+]=[N-])CC2)C1)C(C)C(=O)NC CCC(CC)C(C)C(=O)NCC1CCCCN1C(=O)CCc1cccnc1C c1(C(N2CCC(C)(CNC(CCC#CC)=O)C2)=O)cccc2c1SCCC2 n1(CC)ncc2c(C(=O)OC)ncnc12.c12nc(Cl)c(s1)C(=O)NCC1CCCN21 C1(C(N(C)Cc2ccn(CC)n2)=O)CC2(CCN1C(c1ccsc1Cl)=O)CC2 N1(C(c2[nH]c3cc(C)sc3c2)=O)C2CCCC1CC(NC(C1CCCS1)=O)C2 Cc1nc2cnn(C)c2cc1C(=O)NC(C)CNC(=O)CCN1CCCCCC1 c1(C(=O)OC(C)(C)C)cc(C)n(CCN(C)C)c1C.C(C1CNC(=O)N1)=CC N1(C(C(C2CCOC2)NC(c2nocc2Cl)=O)=O)CCc2nocc2C1 c1(C(N2CCC(CNC(c3cc(C)c(N)cn3)=O)C2)=O)sc2cccnc2c1Cl C(=O)(CC(C)C(=O)N1CC(O)(C2CCCN2C(=O)COCP(C)(C)=O)C1)OC CC1(CNC(=O)CC2CCC2)COCCN(C(c2cc(O)nc(OCF)n2)=O)C1 c1(CC(=O)NC2C(NC(C(C)NC(N)=O)=O)C2)cc2ccccc2c(O)n1 C(=O)(CCC(F)(F)C(F)(F)F)NCC(C)N(C(CC(CC)C1CCC1)=O)C C12(C(=O)NC3(CNC(=O)CCOCC4CC4)CCCC3)CC3CC(CC(C3)C1)C2 N1(SC)CCCN(C(=O)OC(C)(C)C)CC1.c12cccc(c1F)NC(=O)OC2 C1(C)(CNC(CNC(=O)NC)=O)CCCN1C(c1nn[nH]c1Cl)=O c1(C(N(CCNC(C2C(C(C)O)C2)=O)C2CC2)=O)cccc(F)c1O c1(C(=O)NCC(CNC(c2cc(C3CC3)cs2)=O)OC)cc(C)cc(O)n1 n1(CC)cc(Br)c(CC(N2CCCC(CCN3CCCCC3)C2)=O)n1 Cc1c(C(=O)NCc2ccccc2CN(C2CC2(C)Br)C)ncnc1Cl C1(CC(N2CCN(C(C(c3ccc(C)s3)C)=O)CC2)=O)CCOC(C)(C)C1 N1(C(C(CC)OC)=O)CCC(C)(NC(c2csnc2OC)=O)CC1 C(=O)(C1=CCC(C)CC1)N1CCC(C#C)(C(=O)NCC2CC(CN=[N+]=[N-])C2)C1 C1(CNC(C2CC(CCOC)C2)=O)CC2(CC2)CN1C(=O)Cn1c(C)ccc1C c1(CC(CNC(=O)NCC(c2cccs2)O)CO)ccccc1F C1(C(N2C(CN(C)C(c3ccoc3)=O)COCC2)=O)CC2(CCC2OC)C1 N1(C(C2CN(CCC)C(=O)C2)=O)CC(C2CCCCN(C(C3SCCS3)=O)C2)C1 C1(CC(=O)NCC2CC(O)CN2C(c2ccc[nH]2)=O)CCC(=O)NC1 c1(CC)ocnc1CNC(C1(N(C(C2CCCC2CC)=O)C2CC2)CCC1)=O C(=O)(C(CC)(CC)CO)N(C)CC1CCN(C(Cc2ccn(CC)n2)=O)CC1 c1(OCC)ccc(C)cc1C(=O)NC(C)C(c1ccc(Cl)cc1)O c1(OCC)ccc(-n2ccnc2)c(Cl)c1.c12cnc(nc1OC)[nH]c1ncc2s1 C12(C(N(C(C)CNC(=O)CC3CC(O)C34CCC4)C)=O)CCC(CO)(CC1)CC2 C(=O)(C1CCCc2nncn21)NC1CC(CNC(CC(C)SC)=O)C1 C(C#CC1CC1)NC(C=CCN(C)C(C1CCSCC1)=O)=O N1(C(C2C(C)C2C)=O)CCCC2C1CCN2C(c1ccc(C#N)cc1O)=O C(=O)(CN=c1cc[nH]cc1)N1CCC(C(=O)NCC(C)OC)C1(C)C C1(C(=O)NCCCCC(=O)NCC(C)(C)n2cccn2)CC2CC1CC2O C(C)(C(CO)NC(=O)CCCn1cccc1)NC(C(C)OCC=C)=O C=CCCCCC(=O)NC1CN(C(c2cc(Cl)no2)=O)CC1n1cccn1 C1(CC)CCCN(C(=O)Cc2cc(C)no2)C1C(=O)NCC1CC1 N1(C(c2c(NC)snc2C)=O)CCCCC(NC(c2ncccc2Br)=O)C1 c1(C(=O)NCCC(C)NC(C2(CC=C)CCC2)=O)cc(Br)cn1C(C)C CC1CC(C(=O)NCC2(CNC(c3cn4ccsc4n3)=O)CC2)CC(C)C1 n1(CC)c(O)nc2cc(C(N3CCC(NC(=O)CC(C)C)C3C3CC3)=O)ccc12 CC(C)(C(=O)NCCC1CC(NC(=O)C(F)(F)C(O)C2CC2)C1)S(C)(=O)=O C1(C(NOCCOCCOC)=O)(C(C)C)CCCN1C(c1oc(C)nc1C)=O Cc1oc(C)c(C(=O)NCC(C2(O)CN(C(c3cc(O)nn3C)=O)C2)(C)C)c1C CC(O)C(C)NC(=O)C(C)NC(C1CC(OC2CC2)C1)=O C1(CNC(C2C3CN(C(=O)C4=COCCC4)CC23)=O)CC2(CCO1)CC2 C1(O)(C(C)NC2CCCCC2(C)C)CCN(C(=O)NC2CCCC(C)C2)CC1 c1(C(C(=O)N(CC(C)NC(=O)COCCN(C)C)C)C)ccc(Cl)cc1 C(=O)(C(O)CCC(F)(F)F)N1CC2(C(N(C)C(C3C(C)(C)C3(C)C)=O)CCC2)C1 C(=O)(C1=CCCCC1)N(C1C(CNC(CC2(C(=O)OCC)CCC2)=O)CC1)CC N1(C(C(C2CCN(C(c3c(C)ccnc3C)=O)C2)F)=O)CCCN(C)CC1C N1(C(C=CC(C)=O)=O)CC(NC(=O)Cc2nccn2C)CC1C C(C(=O)N(CCC(=O)O)C)(C(C)(C)C)c1cn(C2CCC(N(C)C)CC2)nn1 N1(C(c2c(COC)cco2)=O)CCCC(NC(=O)CN(S(C)(=O)=O)C)CC1 c1(C(=O)NC(CNC(CC(C)F)=O)C2CC2)cc(Br)cc(-c2nn[nH]n2)c1F N1(C(C(N)=O)=O)CCc2sccc2C1CNC(c1cc2c(O)cccc2[nH]1)=O C(C1=CCN(C(C2(F)CCOCC2)=O)CC1)NC(C(C1CCCC1)OC)=O C1(CNC(c2nn(CC)c(C3CC3)c2)=O)CC(C)(C)CN1C(C1CCC1OC)=O c1(SCC(N2CCCN(C(C3C(OC)CCC3)=O)CC2)=O)ncnc2[nH]cnc12 C1(NC(C2CN(C(C(C)SCCCC)=O)CC23CC3)=O)CCC2(CCCC2)C1 C(=O)(CC=C(Cl)Cl)NC(C)CC1CN(C(=O)COCCc2cnccn2)C1 Cc1cc(C(=O)NC2CC(C(F)C(=O)NCC=C(Cl)Cl)C2)c(C)o1 C1(C(=O)NCCC2C(C)CCC2)C2CC1N(C(c1ccc(O)nn1)=O)C2 Cc1nscc1CC(=O)NC1(C(N2CCC2(C)C(=O)N(C)C)=O)CCCC1 CC1CC(=O)NC(C(=O)NC2CC3CC2CC3C(=O)NCCN2CCCCC2)C1 CC1CN(C(=O)CCC2CC2C)CC1(C)C(=O)N(C1CC2CCC1CC2)C C1(NC(c2[nH]cc(C#N)c2)=O)CC2CCC1CC2NC(C1CC1Cl)=O c1(Nc2ccc(C)cc2)c(Br)cncc1[N+](=O)[O-].C12COCCN(C1)CC(=O)N2 C1(CN(C(COCC(=O)NC)=O)C)CCN(C(=O)C(C(C)C)SCC(C)C)CC1 C1(C)(CNC(CCCOC(C)=O)=O)CCN(C(c2ncnc(O)c2F)=O)CC1 c1(NC(N(C2(OCC)CCCC2)CC)=O)ccc(SC)c2ccncc12.C(C)(C)(C)O c1(C(=O)NC2C(NC(c3cc(C)n(CCO)n3)=O)COCC2)c(F)cccc1F N1(CCC)CCN(C(=O)C(C#N)NCCCn2ccnc2C)C(CC)C1.C1CC1 CC1CCC(C(=O)NC2COCC2O)N1C(c1cnc[nH]1)=O c1(OC)c(C(c2nnnn2CCCSC)Nc2ccc(C)cc2)cccc1Cl C1(C(=O)NC(CCCNC(C(C=C)(C)C)=O)c2ccccc2)CCC(=O)N(CC)C1 O(NC(=O)C(CNC(=O)CCCC(F)(F)F)CC1CC1)C(C)C c1(C(N2CCC(O)(CSC)C2)C(=O)NCCCC)ccc(OC)c(OC(F)F)c1 c1(CN2C(C(=O)NCCSC)C3CCC2C3)ccc2c(c1C)OCCO2 C1(C(=O)NCC(COCC)(F)F)CN(C(C2CCC2CO)=O)C(C)(C)C1 c1(C(=O)NCC#CCNC(C(C)OCC#C)=O)cc2sc(Br)cc2s1 C(CC(=O)NC1CC(C(F)C(=O)NCCOCC)C1)SCCCC c1(OCC=C)ccc(Cl)c(C(=O)NCC2CN(C(c3cnsc3)=O)C(C)(C)C2)n1 C(CC(=O)NC(C)CNC(c1cc(F)c(F)c(F)c1O)=O)(C1=CCCC1)OCC c1(CC)cccc(CNC(N2CCC(NC(C3CC3(F)F)=O)CC2)=O)c1 N1(C(CCC)=O)CCC(O)(C2CCN(C(=O)C(COC)OC)CC2)C1 N1(C(c2n(CC)ccc2)=O)CC2(CCC2CNC(C2CC3CCC2O3)=O)C1 N1(CC(=O)N(C2CCN(C(C3CCN(CC)C3)=O)C2)C)CCN(C)C(=O)C1 C#Cc1ccc(C(=O)NC(C)CNC(c2sccc2CC)=O)nc1 c1(C(N2C(CNC(c3c(Cl)cc(C)s3)=O)C(C)CC2)=O)cccc2c1C(=O)NC2 C1(COC)(NC(=O)C(=O)NC2CC2)CCN(c2ccnc(C)n2)C1 C1N=C(N2CCC(SC)C2)NC(C)Cn2nccc21.c1(CC)ccccc1F C1(NC(C(CCC)CC)=O)CC2CCC(C1)N2C(=O)C(F)CCC(C)C C1(C(=O)NC(C)CCN(C)C(C2CC3CC2C3)=O)(NC(C)=O)CCCC1 C1(C(=O)NCc2nc(C(C)(F)F)sc2)CC2C3C=CC(C3)C12 C(=O)(CC(C)(F)F)C(CCCc1ccc(SC)s1)=O.C1(NC)CCNC1 C1(CC(=O)N(C2CCCC(NC(c3n[nH]c(C)c3Cl)=O)C2)C)CC(=O)NC(=O)C1 c1(N2CCCC(CNC(c3ccc(Cl)o3)=O)C2)nc(Cl)nc2ccc(Cl)nc12 CC1=C(C(=O)N2CC=CC2CNC(c2c[nH]nc2F)=O)Cc2ccccc2O1 N1(C(C(C)OCC#C)=O)CC2(CCC(NC(c3cc(=O)cc[nH]3)=O)CC2)C1 CC(CCOc1ccccc1)C(=O)NC1CC(NC(=O)C(F)C2CCCC2)C1 c1(OC)ncnc(C(N2CC(O)(CCNC(c3cccc(O)c3Cl)=O)C2)=O)c1F c1(C(=O)NCCC(C)NC(=O)Cc2cc[nH]c2)ccc(Br)c([N+](=O)[O-])c1 c1(CN2CCC=C(C(=O)NCCNC(C)=O)C2)cc(Br)c2cc[nH]c2c1 C12CCCC1(c1nnnn1CCCF)NCC2.c1(C)ccoc1.CN(C)C(N)=O c1(C(=O)OC)ccc(N2CCN(C3CCCC(C)C3)CC2)nc1 C1(C(=O)NC(C2(C(=O)NC(C34CCC(CO3)C4)C)CC2)C)CC2C=CC1C2 CC1(C)C(C(=O)NC2CCN(C(C34CCC(CC3)C4)=O)C2C2CC2)CCS1(=O)=O N1(C(CCCN(C)C)=O)CCC2OCCN(C(C3CC4CC3CC4O)=O)C2C1 N1(C(C(CCSC)O)=O)CCN(C(=O)CC2(C)CCCC2)CCC2(CC2)C1 C(=O)(C1CCc2nccn21)NC(C1CN(C(C(C(C)C)NC(N)=O)=O)C1)C C(=O)(CCCCCc1ccccc1)N(C(CC)CNC(=O)CCC(=O)NC)CC c1(C(=O)NCCC(NOCCCC#C)=O)cc2cccnc2[nH]1 CC(CC(F)(F)F)C(=O)N1CCCCCCC1C(N1CCC(C)(C)C1C)=O N1(C(c2c(C)n(C)cc2)=O)CC2CC(C1)N(C(=O)C(O)CC1CCCCC1)C2 N1(C(Cn2cc(C3(COC)CCOCC3)nn2)=O)CC(C(N)=O)CC(C)C1 c1(C(N2CCC(C)(NC(c3ccc(OCC)cc3)=O)C2)=O)coc(S(N)(=O)=O)c1 c1(NC(CC(C)NC(C2(C)COC(=O)N2)=O)=O)cn(C)nc1C#N Cn1ccc(-c2cc(C(=O)N(c3cnn(CCc4nn[nH]n4)c3)C3CC3)no2)n1 C(C(C)(C(=O)NCc1cscn1)NC(=O)CCC1CCC(=O)C1)SC C#CC1(C(=O)NCCC(C)C)CCN(C(=O)CSCc2ccccn2)C1 C1(NC(CCC(=O)NCC)=O)CCN(C(c2ccnn2C2CCC2)=O)CC1O N1(Cc2ccc(N(C)CCO)cc2)CCC2(CCC(O)C2)C1.N12CCCC1C2 N1(C(COC)=O)CCN(C(c2ccc(-c3ccccc3)cc2O)=O)CC1CF C1(NC(c2cc(COC)on2)=O)CCCC(C(=O)NC2CC2c2ccco2)CC1 C1(NC(C(=Cc2cnc[nH]2)C)=O)CCCC(NC(c2ccsc2C)=O)CC1 c1(CC(=O)NC2C(CN(C(c3cc(C)sc3N)=O)C)CCC2)c(C)ncnc1C n1(CCC(=O)NCC2CN(C(CC=C)=O)CC2F)cc(S(N)(=O)=O)cn1 CCC(C)CCC(=O)NC(C)C(=O)NCc1cccc(OC)c1 C(C)(C)(CC(=O)NC1CN(C2CCC2)C1)N(C(c1c(OC)csc1)=O)C C12(C(N3CCCC(CN(C(c4ccccc4O)C)C)C3)=O)CCCC1C2(F)F C1(OC)CN(C(=O)Cc2cnn(C3CC3)c2)CC1NC(=O)CCC#N C12(CNC(c3cc(OC)ns3)=O)CC(CN1C(C1CC(C)OC1C)=O)C2 c1(C(=O)NC2CC(C(C)NC(c3cnc(C)o3)=O)C2)nccnc1C N1(C(CSCC(C)C)=O)CCC(O)(CCNC(C2CNC(=O)CC2C)=O)CC1 C1(NC(N2CCC3(C(C(=O)OC)C3)CC2)=O)CCCCC12CCCCC2 n1(CCC(=O)NC2CCN(C(C(CCCC)O)=O)C(C)C2)cnc2ccccc12 CC1CC(C(N2CC=CC2(C)C(=O)N(C)C)=O)CN(C(=O)CCCC(=O)N(C)C)C1 C(=O)(C#CC1CCCCC1)NC1CCN(C(CSCC(C)C)=O)C1C N#Cc1cccc(C2CC2C(=O)NCC(O)CNC(=O)Cn2ncnn2)c1 C(CCCCCN(C(=O)Cc1ccsc1)C)NC(C(=O)NCCOC)=O C1(C(=O)NCC(=C)CCNC(c2cnnc(C3CC3)c2)=O)CC(=O)NC(C)C1 C(=O)(C1CCCc2cc(C#N)ccc21)NC1CC(NC(C(CC=C)(C)C)=O)C1 CC(CN(C)C)CCC(=O)N(CCCNC(c1ccnc(N(C)C)c1)=O)C C(C)(C(C)C(=O)NCCN(C1CCCC1)C)NC(C=C(CC)CC)=O C(=O)(C(=O)CC(C)CC)N1C(CC=C)(C(=O)NCCc2ncccn2)CCC1 C(=O)(C1=COCC1)N1CC(O)(C(C(=O)NC(C2CCC(=O)N2)C)F)C1 N1(C(C2(C)N(C(C)=O)CCC2)=O)CC(NC(=O)C2=NOCC2)CC(F)(F)C1 N1(C(C(OCC)C2CC2)=O)CC(C)(NC(=O)COc2ccc(C)cc2F)CC1(C)C c1(SC)cc(C(=O)NCCC(C)N(C)C(c2c(C)noc2N)=O)ccn1 C1(NC(COCP(C)(C)=O)=O)CC2CC1N(C(c1coc(C3CC3)n1)=O)C2 Cc1csc(=Nc2ccc(Cl)cc2)n1CCC1CC(C)(C)OC(C)(C)C1 c1(NC(CCCN(C(C2C(CC(C)C)C2)=O)C)=O)ccc(OCC(F)(F)F)cc1 C(=O)(C1=CCCCO1)NC1CCN(C(C2(N(C)C)CC2)=O)C1c1ccccc1 c1(CNc2cn(C)c(C(=O)Nc3ncc4[nH]ncc4n3)n2)c[nH]c2ccccc12 C1(CNC(CCn2ncn(C)c2=O)=O)CN(C(=O)C2=COCCC2)CC12CC2 c1(CNC(C2(CC=C)CN(C(c3ccon3)=O)C2)=O)nc(C)c(C)s1 C=CCC(CNC(=O)CC1(O)CCC1)C(=O)NCc1cncc(OC)c1 C1(C(N2CCC(C)C2CNC(=O)COC2CCOCC2)=O)CCC2(CCC2)O1 C#CCC(CC(=O)N1CC(n2cnnn2)C1)NC(=O)CN(CC)CC O=C1NCc2cc(CNC3CCCN(S(=O)(=O)c4cnoc4)C3)ccc21 CCC(C)CCCC(=O)N(C)CC1CCCN1C(c1cc(F)cs1)=O c1(C(C)(C)C)n[nH]c(=NC2CC(NC(=O)COCc3cccc(Cl)c3)C2)o1 C(=O)(C(C)CC(C)(C)C)N1C(C)CCC(NC(C(C)=C(C)C)=O)C1 c1(NCC(C)(C)NC(=O)C(O)CC2CCCCC2)nc2c(cc1C#N)CCCC2 CC1(C)CC(NC(c2ccc(=N)[nH]n2)=O)CN1C(c1csc(Br)n1)=O C(=O)(C(C)(F)C(=O)N1CC2CC2(NC(=O)CNC=O)C1)OC C(=O)(C(CCC1CCC1)NC(=O)CCN=[N+]=[N-])N1C(CN=[N+]=[N-])CCC1 N1(C(C(=O)N(C)C)=O)C2CCC(C2)C1C(=O)NC1CC2CCCC2C1 Cc1cc(CC(N2CC3CC2CC3NC(c2coc(C(N)=O)c2)=O)=O)cc(C)c1 c1(C(N(CC(C)(C)CNC(=O)CCC2CC2(F)F)C)=O)ccc2nc(O)oc2c1 N1(Cc2c(O)cc(Br)cn2)c2ccccc2SC2CCCC12 c1(OCCC(=O)NC(CNC(CC(C)CF)=O)C(C)C)ccc2c(c1)CCCC2 c1(C(N2CCCCC(NC(C(C)S(C)(=O)=O)=O)C2)=O)ccc2c(c1)COB2O C1(NC(C(C2CCN(C(CCCN(C)C)=O)C2)F)=O)CCC(C)(O)CC1 N1(C(C(C)NC(CC)=O)=O)CCCc2n[nH]cc21 CCC(CCOC)C(=O)NNC(=O)C(C)(C)CCCCNC(C1CC(F)C1)=O O=C1COC(CNC(c2ccc(NC(c3ccoc3)=O)nc2)=O)CN1 c1(C(N(CCNC(Cc2ccc(C)nc2)=O)C)=O)n[nH]c2ccc(F)cc12 C1(CNC(c2ccccn2)=O)CN(C(C2C=CCCC2)=O)CCC1C(F)(F)F C1(CCC=C)CCCN(C(CCC2CC2)C(=O)NCc2nnn(C)n2)C1 C1(C)(C(=O)NCN(C)CCOCCC(=O)NC2CNC(=O)CO2)CCCN(C)C1 C(C)(CC(C)C#N)(c1n(-c2c(C)cccc2)nnn1)N(CC)Cc1cc(C#N)cs1 C12(COCC)CC(NC(C3(NC(c4cnoc4)=O)CCC3)=O)(CO1)C2 c1(NC(C(=O)OCC)=O)ccc(NC(=O)C(=O)NC2CC(N(C)C)C2)c(C2CC2)c1 CC(CCC(C)(C)C)C(=O)NC1(CO)CCCN(C(=O)C=CS(F)(F)(F)(F)F)C1 C1(NC(C2(C)C=CCCC2)=O)CN(C(=O)COCC2CCOCC2)CC1(C)C CCCCC(C)CC(=O)N1CCN(C(C2CCN(CCC)CC2)=O)CC1CCC C(C(F)(C(=O)NC1(c2cccs2)CC1)C(C)C)NC(C(CC=C)CC)=O N1(C(CSCC)=O)CCC(C2CCCN(C(=O)C3CCCn4ccnc43)C2)CC1 C1(C(N2CC(N(C(=O)CCc3nc(=N)[nH][nH]3)C)C2)=O)CC(C)(C)OC1(C)C N1(C(CCC=C)=O)CC2CC(NC(=O)CCOc3cccc(C)c3C)C1C2 C(=O)(C(CO)C(F)(F)F)N1CC(CCC)C(C(=O)NCC(C)OC)C1 C(=O)(CC(F)(F)C(F)F)NC1C2(CC(NC(Cc3n(CC)nc(C)c3)=O)C2)C1 c1(CC(=O)NC(C2CCN(C(c3cc(N)cnc3Cl)=O)C2)C)ccn(C)c(=O)c1 c1(C(=O)NC2CCN(C(c3n(C)nc(C(C)(C)C)c3)=O)C2)n[nH]c2cccnc12 C(C1=CCN(C(c2cc(C)ccn2)=O)CC1)NC(C(C)NC(COC)=O)=O C1(CCNC(C2(CCOC)SCCCS2)=O)CN(C(=O)CSC)CC(C)O1.C(C)=O C1(CNC(c2cc(C)ns2)=O)CN(C(C2CC2c2nc[nH]n2)=O)CC1(C)C C(CC(C)NC(=O)CNC(=O)OC)NC(COCCOC)=O CN1CC(C(=O)NCC(CO)NC(=O)CCF)c2ccccc2C1=O C1(CN(C(CC2C(CC)C2)=O)C)CCCCN1C(=O)COCC1CC1 c1(OC)cnc(CNC(=NCC2CCOC(C)C2)NCCN2CCOCC2)cn1 CC(C)(C)CC(O)CC(=O)NCCN(C1CCCCC1)C(C1C2(CC2)C12CC2)=O c1(CC(N2C(COCCCOC)CCCC2)=O)cc([N+](=O)[O-])cc2c1OCOC2 C(=O)(N=c1cc(C)[nH][nH]1)C1C2CN(C(C(CC)(C)O)=O)CC1CC2 N1(C(CC2N(CC)C(=O)CC2)=O)CC2C3CCC(C2C1)N(C(=O)C=CCOC)C3 C1(CC(=O)N(CCN2CCS(=O)CC2)C2CC2)CCC2COCCC2O1 O=C(CC1COCc2ccccc21)NC1CCC(F)(CNC(=O)C(F)F)C1 N#Cc1ccc(O)c(C(=O)NCC2CCCCN(C(=O)C(F)=CCCF)C2)c1 c1(C(=O)NCC(CC)NC(c2cnc(SC3CC3)n2C)=O)cncc(NC)n1 CC1CCN(C(=O)C(N2CCCC(CN(C(=O)COCC(F)F)C)C2)=O)CC1 CC1CC(C)(C(N2C3CCC2CC(NC(=O)CCNC(N)=O)C3)=O)CC(C)O1 CC(CN(C)C(c1cc(O)cc(=O)o1)=O)C(=O)N1CC2COCC2O1 c1(N2C(CNC(c3nc(COC)sc3)=O)C(C)CC2)nc(OC)cc(C)n1 c1(C(N(C2CCCC(NC(c3ncc(F)cc3N)=O)C2)C)=O)ccc(F)cc1Cl C(=O)(CCCCCCNC(=O)Cn1cc(CO)nn1)N(C(C)C(N)=O)CC N1(C(C(CC=C)C(C)C)=O)CCC2CN(C(c3n[nH]cc3Cl)=O)CC2C1 C1(C(=O)NCC2N(C(c3ccnc(C)c3N)=O)CC2)CCc2ccccc2O1 N(C(=NCCF)N1CCC2C(C(N)=O)C2C1)CC(C)C(=O)N1CCOCC1 CC1CCCN(c2cncc(Cl)n2)C1C c1(CC)c[nH]c2ncnc(NCC(CC)NC(C3(C)CC3)=O)c12 C1(C(=O)NNC=O)CN(CCc2ccccc2)CCC1O.NC=O c1(C(=O)NC2(CNC(C(CC)O)=O)CCOC2)cccc(NCC2CC2)c1 C1(C(=O)NC(CN(C(=O)CC23CC(C2)C3)C)(C)C)CCCOC1 C1(CNC(C2(CC#C)CC2)=O)CCCCC1NC(C1(F)CCOCC1)=O CC1CCN(C(=O)C(C)(C)C)CCN1C(C1CC(=C(F)F)C1)=O CCC(C)(C)C(O)C(=O)N1C(CC(N2CC3CC2CC3O)=O)C2CCCC12 c1(C(N2CCCC2C2CCN(C(=O)C=C(CC)CC)C2)=O)cc(OC)c(C)o1 c1(C(=O)NC2C(CNC(CC(C)F)=O)C2)ccc(C(F)(F)F)cc1C(F)(F)F C(=O)(CCCN=c1nc(N2CCC=C(Cl)C2)c2c(ncn2C)[nH]1)N(C)C C(=O)(C(C)S(=O)(=O)C(C)C)N1CC(CNC(C(C)=C2CC2)=O)C(C)(C)C1 N1(C(CN(CC)CC)=O)CCN(C(=O)Cc2cc(CC3CC3)on2)CC(O)C1 N1(C(c2c(C)n(C3CC3)cc2)=O)CCC(NC(c2ccoc2Cl)=O)C2(CCC2)C1 CC(C)CC(O)C(C)C(=O)NC1CC2(C1)CN(C(=O)Cc1csnn1)C2 N1(C(C(C)CN(C)C)=O)CCN(C)C(C(=O)Nc2cccnc2S)C1 N1(C(C(CC#C)NC(C2CCC2COC)=O)=O)CCC(N(C)OC)CC1 c1(N(C)C)cccc(=NC2CC2CS(N)(=O)=O)[nH]1 C(=O)(CCC(CF)CF)N1C(C(=O)NC(CCN(C)C)(C)C)CC1 C(N=c1nc(N2CC=CCC(C)(C)C2)c2sccc2[nH]1)c1n(C(C)C2CC2)cnc1 c1(NCC(C(C)C)N(C)C)ncc(S(=O)(=O)NCC2CC2)cc1Cl CC1CC(c2ccccc2)CN1Cc1cc(-c2cccc(OC3CC3)c2)no1 CS(=O)CCC(O)C(=O)NCC(CO)(CO)NC(=O)CC1(O)CCC1 C(=O)(C(F)(F)CN1CCCC1)N(C1CN(C(=O)C(c2ccccc2Cl)O)C1)C N1(C(C=C(C)C)=O)CC2CC(NC(c3ocnc3C)=O)CC2C1 c1(CCC)noc(CCCNC(c2nnnn2CC(F)F)c2ccccc2)n1 c1(CC(C)C)n[nH]cc1C(c1nnnn1C1CC1)NCC(C)(C)C1CC1 Cc1nn(C)c(Cl)c1C(=O)NCCCN1CCC(NC(C2(C#N)CCSCC2)=O)C1 Cc1cc(C(N2CCC(C3CCCN3C(C3CC(C#N)C3)=O)CC2)=O)n(C)n1 c1(C(N2C(CCNC(c3cocn3)=O)CSCC2)=O)coc2cc(F)ccc12 C1(NC(=O)C(F)OC(F)(F)F)CCN(C(=O)CN2CC3CCC2C3)C12CC2 C(CO)(C(=O)NCC1CCN(C(=O)CC2CC2)C1)NC(C(C)C)=O c1(NC2CC(CNC(=O)CC(c3cccc(F)c3)O)C2)ccc([N+](=O)[O-])cn1 [N-]=[N+]=NCCCCNC(C1C=CC(NC(c2ccc[nH]2)=O)C1)=O c1(NCC(C(C)(C)C)OC)ncccc1S(=O)(=O)NCCCSCC(C)C c1(CN2CC(C#N)C(Nc3ncnc4c(Br)c[nH]c34)C2)cccc(Br)c1[N+](=O)[O-] CCC(CC(=O)NCCCCOC)NC(C1(N2CCNC2=O)CC1)=O c1(C(=O)NC2(CCNC(Cc3c(C)ncs3)=O)CC2)cc(F)c2[nH]nnc2c1 C(C1=NOC2CN(C(=O)COCc3nc[nH]n3)CC12)NC(c1c(C)cc(F)s1)=O N1(C(CCN(CCC)C)=O)CCCCC(NC(c2cnnn2C(C)C)=O)C1 c1(C(=O)NC2CCCC(NC(c3n(CC)ncc3)=O)C2)nnc(O)c(Br)c1O C(C(O)C(=O)NC1CCC(CCC(=O)NCc2ncsc2C)C1)SC c1(NC(C2N(C(c3[nH]cc(C)c3)=O)CCSC2)=O)ccc([N+](=O)[O-])c(C)c1 Cc1n[nH]c(=NC(C)C2CCCCN2C(c2cnc3c(c2)COC3)=O)s1 N#Cc1cc(CN2CCOCC(C(N3CCC(C4CC4)CC3)=O)C2)cc(Cl)c1 CN=c1nc(N2Cc3cc(OC)ccc3C2)[nH]c(=NCCCc2n[nH]c(=N)s2)[nH]1 N1(C(C(c2ccc(CC)cc2)C)=O)CCC2C(C1)CN2C(=O)COc1ccsn1 c1(CNCC2(NC(c3n(C)ccc3)=O)COC2)c(F)cc(Cl)cc1Br N1(C(C(CSC)O)=O)CCC2(CC1)CC(NC(=O)C(C)OCc1ccccc1)C2 C(C(C)(C)C#CC(=O)NCCCn1ccnn1)NC(C(C)CC(N)=O)=O c1(OC)ccc(C(=O)N(C)Cc2cc(C(=O)NC(C)CO)ccn2)cc1 CC(C)S(=O)(=O)CC(=O)N1CCCC(C2(C(F)(F)F)N=N2)C1.C1CO1 c1(C(C)NCC#CCOC)cc(F)ccc1OCc1ccccc1 N1(C(COC2(C)CCOCC2)=O)CCC2(CCCCC2NC(=O)CSC2CC2)C1 Cc1cc(Br)oc1C(N1CCC(CCNC(=O)CN2CCC(O)CC2)C1)=O N1(C(C(=O)NCC)=O)CC(NC(c2cc(C(F)F)ccc2OCC)=O)CCC1C c1(C(=O)NCC2C(NC(c3ncn(C)c3)=O)CCC2)c(F)ccc(O)c1F c1(NC(=O)NCC2(C)ON=C(C)C2)c(O)nc(=O)n2c1CCC2 C(F)(C(F)(F)F)(C(F)(F)F)c1ccc(C(C2(c3cncnc3)CCOCC2)=O)cc1 CC1CCc2onc(C(N3CC4CCN(C(C5CS(=O)(=O)C5)=O)CC4C3)=O)c2C1 C1(NC(c2csc(-c3ccoc3)n2)=O)CCN(C(=O)C(F)CC2CCC2)CC1F N1(C(C2CC=CC(NC(C3N(C)CC3)=O)C2)=O)CCCCC(C)(F)C1 n1(CC(=O)NC(CCNC(CC2CC(OCC)C2)=O)C)cnc2ccc(C)cc12 CCCC(CNC(C1(CC)CCCC1)=O)C(=O)NC1CCCCC1C(=O)OC N1(C(c2cn(C)nc2)=O)CCC(NC(C2(C)C=CCC2)=O)C(O)C1 c1(C(=O)NC2CCCN(C(c3c(CC)nco3)=O)C2)ccc2c(c1)C(=O)CCN2 CCN=C(NCCc1cccc(F)c1)NCCN1CCCC1C c1(NC(C2CC(C)(NC(=O)CCn3ccnc3)C2)=O)ccccc1C1CC1 C1(NC(C(CC=C)C)=O)CN(C(=O)C(c2cnc(O)nc2O)(F)F)CC12CC2 CC(C)C(F)(CNC(=O)C(C)C1CCC(=N)N1)C(=O)Nc1cccc(N(C)C)c1 C1(C(=O)NCCN(C(C)C)C(C2CCOCC2)=O)CCC(=O)CC1C c1(C(=O)NCC(CNC(C(c2ccc(Cl)cc2)OC)=O)F)cn2c(n1)CCCC2 C12CN(CC(C)(C)O1)C2=O.CCCCC(O)C(=O)NCC1(c2ccncc2)CC1 c1(C(N2CC(CN(C)C(C34CC3C4)=O)OCC2)=O)ccc2c(c1)C(=O)NC2=O n1(CCC(=O)N(C2CCN(C(CC(C)c3cccnc3)=O)C2)C)cnccc1=O c1(C(N2CC(CNC(C(=O)NCCOC)=O)C(O)C2)=O)cc([N+](=O)[O-])cnc1O CCCC(C)C(=O)NCCC(C)(C)CNC(=O)C(C)CCOC C1(NC(=O)C(CO)c2ccccc2)CCN(C(c2cnc(Cl)s2)=O)CC1 C1(C(=O)NCCC(C)NC(=O)CC2(O)CCCOC2)(CO)CC2CCC1CC2 N1(C(=O)N(c2cnc(C)s2)C)CCCC(N(C(=O)OC(C)(C)C)CC)C1 C(CCCCCC(=O)NC1(c2ncccn2)CC1)NC(c1c(C)n(C)cc1)=O C1(C(N(C2CCC(NC(C3CCN(C(=O)OCC)C3)=O)C2)C)=O)CC2C=CC1O2 C1(C(=O)NCC2(NC(COCC)=O)CC2)CCC(CC)C1 C(CC(C)C(=O)N1CCC(N(c2ncc(OCC)cn2)CC)C1)=CCC N1(C(C(C)NC(COC)=O)=O)CCCC1C(C)NC(c1coc(C(F)F)n1)=O CC(C)(C)CCCCC(=O)NCCOCCNCC.S(C)(=O)(=O)NCCO Cc1cc(C(N2CCCOC(CNC(=O)C3=CCOC3)C2)=O)c(C)n1NC(N)=O c1(CC(=O)NC(C2CCCN(C(C3(Cl)CC3)=O)C2)C)ccc2nonc2c1 C12(NC(C(C)CN(C)C)=O)CCCC1CN(C(=O)CCC(=O)N(C)C)C2 C1(COC)(NC(C2CC3(CC3)C2)=O)CCN(C(c2coc(N(C)C)n2)=O)C1 C(=O)(CCCF)NC1C(CC(=O)N(CC=C)CC)C1 CC1(C)CC(NC(c2csc(CO)n2)=O)CN1C(C1(C2CCC2)CC1)=O CCCCS(=O)(=O)N1C2CN(C(c3ccccc3C)=O)CC12 c1(CC)nnc2cc(NC3CCCC3NC(c3cn4cccnc4n3)=O)ncn12 N1(C(c2ccc(-n3cnnn3)cn2)=O)CCC2(CC(NC(C3CC(O)C3)=O)C2)C1 Cc1ncc2n1CCN(C(C1CCN(C(=O)CC34CCCC3C4)O1)=O)C2 c1(C(=O)NC2(C)CN(C(CCC=C(C)C)=O)C2)cnn(CC(C)C)c1C c1(C(N(C)CC2N(C(c3c(C)nnn3C)=O)CCCC2)=O)cnn2ccn(C)c12 N1(C(c2cnc[nH]2)=O)CC(C2CCN(C(=O)CCN)C2)C1.N1(C=O)CCCS1(=O)=O N1(C(CSCC#C)=O)CC2(NC(=O)CSSC)CC1C2 Cc1nc(O)nc(C)c1C(=O)NCC1CCCCC1NC(=O)C(=O)N1CCCC1 C12(CNC(c3c(COC)cccn3)=O)CCCCC1CN(C(=O)C=CC1CC1)C2 C1(C(=O)OC)CCCN(Cc2n[nH]c(-c3ccccc3)n2)C1CN(C)C N1(C(=O)NC(C2CCOC2)C)CCN2CCC1C2.c1(C2CC2)cn(C)nn1 c12cc(C#N)c(nc1C)SC2.C=CC(O)C(=O)NC1CC(NC(=O)C=C2CC2)C1 CS(=O)(=O)c1ccc(CN2CCC(n3cc(C4CCCC(F)(F)C4)nn3)CC2)o1 C1(C(=O)NC2(C(=O)NCC3CC(CC)C3)CCCC2)COCC(C)O1 n1(CCNC(C(C2CCN(C(CC)=O)C2)C)=O)nc(C)cc1C N1(C(C(CC#C)O)=O)CCC(C=CC(N2CCN(CCF)CC2)=O)CC1 N1(C(COCC)=O)CCC2(CC1)CN(C(c1ncncc1Cl)=O)C1COCC21 c1(CCC)nc(C)c(C(=O)N(C2CCN(CCF)CC2)CC)o1.C1(C(=O)N)CC1CC N1(C(CCNC(=O)CO)=O)CC(CNC(=O)C(C2CCCCC2)O)C(F)C1 N1(C(c2c(C)cn(C)n2)=O)CC2CC(Nc3ccc([N+](=O)[O-])cn3)CC1C2 c1(NC(CC2CCN(c3nccc(C)n3)CC2)=O)cc(Cl)cc(Cl)c1O c1(-c2n(CCC(C)C)nc(-c3ccc4c(c3)CCC4)n2)cnc2cnn(C)c2c1 C1(CSC)CCC(N=c2nc3cnn(C)c3c(N3CC4C(C3)C4(F)F)[nH]2)C1 N1(C(c2ccc(C)c(C)c2)C(=O)NC)CC(SC)C(C2CC2)C1 CC(C)(C)CCC(F)C(=O)N1CC2CC1C2NC(c1cc(C(N)=O)c[nH]1)=O C(=O)(CCCC(=O)NC(C)C)NC(CCCC)CNC(=O)CN(C)C N1(C(=O)Nc2cn(CC=C)nc2)CCS(=N)(=O)C(C)C1 Cc1sc(O)nc1C(=O)NCC(C)(O)CNC(=O)C=C1CCC1 Cc1ccc(C(=O)NCCCCCNC(=O)CCCOc2ccccc2)cc1 C(=O)(C(=O)NOCC(OC)OC)NC(CCC)C1CCCC1.OC CCC(C)CC(=O)C(=O)N1CCC(C2CC2)C1CNC(c1cnc2n1CCC2)=O CCCCC(CNC(C1(NC(C)=O)CCC1)=O)NC(C1CCN(C)C1=O)=O Cc1c(C(N2CC(NC(c3nn[nH]c3Cl)=O)C(C)C2)=O)ccc(F)c1F CC1(C)CCN(C(=O)C(=O)NCC(F)F)C1C(=O)NCC1CCC(C)(C)O1 CC1(C)CN(C(c2ccc3c(c2)CC3)=O)CCC1C(N1CC(N=[N+]=[N-])C1)=O c1(NC(C23C(CN(C(Cc4cc(CC)no4)=O)C2)C3)=O)c(C)nc(C)nc1C C1(C(=O)NCc2cncc(CC(=O)NC(CCC=CC)C)c2)CCOC(=O)CC1 N1(C(C2CCC(N(C)C)C2)=O)CCC(NC(=O)CCOC2CC2)C1C1CC1 N1(c2n(CC(OCC)OCC)c(C(F)F)nn2)CCC(S(=O)(=O)N2CCCC2)C1 c1(COC)ncc(C(=O)NC2CN(C(=O)CCP(C)(C)=O)CC2C)c(O)n1 C12(C(=O)NCCOCCNC(=O)CC3CCOC3=O)CCCCC1C2(F)F n1(CC(N2CCC(C(C(=O)NCC3CN(CC)C3)(C)C)C2)=O)c(C)ccc1C.C1(C)CC1 CN1CC(=O)N(CC(N2CC3CC3(CNC(=O)CSc3nccn3C)C2)=O)C1=O C1(F)(C(=O)NCCOCCC(C)C)CN(C(c2cc(Cl)no2)=O)C1 c1(CNC2CC(NC(c3ccc(O)nc3)=O)C2)ncc(Br)cc1Br C(=O)(CCCSc1cccs1)N(C1CCN(C(=O)C(O)CF)C1)CC c1(C(N2CC(NC(c3c(C)nc(CCC)o3)=O)C2)=O)cnc2c(F)cccc2c1 C1(CNC(c2c(NCC)scn2)=O)CC2CCC1N2C(=O)CCS(N)(=O)=O C(=O)(C(CC(C)C)NC(C)=O)NC1(CC)CCN(C(C2C=CC=CC=C2)=O)C1 c1(C(C)(C)C)cc(CC(=O)NC(C)(C)CNC(C2(n3cnnn3)CC2)=O)no1 CCCC(C(=O)NOCC=CCl)NNCC.C1(=O)C(SCC)C1(C)C N1(C(c2cnn(C)n2)=O)CC2(CCN(C(=O)CCc3ccc(F)nc3)CC2)C1 c1(C(N2CCC(COC)CC2)=O)c[nH]c2c(Cl)cccc12 C(=O)(CC(O)CN(C)C)NC(C1(O)CN(C(c2c(SC)csc2)=O)C1)C N1(C(c2[nH]cc(CC)c2)=O)CCCCC1C(C)NC(c1nocc1Br)=O C(=O)(CC(C)CC(=O)OC)NC(CC(N1CCC(C#C)C1)=O)C c1(C(N(C)CC2N(C(c3cn(CC=C)nn3)=O)CCC2)=O)c(C)coc1CC C1(NC(c2cc(Br)c[nH]2)=O)(CO)CCCN(Cc2ccnc(O)c2)C1 C1(CC(N2CC(CCNC(C(C=C)c3ccccc3)=O)C2)=O)CCC(F)(F)CO1 CC(c1cccc(Cl)c1)=CC(=O)N(C1CN(C(=O)CC2OCCOC2(C)C)C1)C C(=O)(C(C(C)CC)C1CC1)N(CCCNC(c1cc(C)sc1C)=O)CCC C(=O)(C(CCCOC)NC(=O)C1=C(Cl)CCC1)NC(CCC=C)(C)C C1(NC(C2(C)CCC(C)CC2)=O)CCC2CN(C(=O)C(C)(C)O)CCC2C1 c1(C(=O)NC2C(NC(C3(COC)CCC(=O)N3)=O)COC2)cnc2ccccn12 c1(C(=O)NCC(CNC(c2nccc(N)c2)=O)O)cccc2sccc12 c1(OC)ccc2c(c1)OCC(C(=O)N1CC(NC(=O)CC3CCCCN3C)C1)=C2 c1(N(CCCNC(C2CCC(C)CC2)=O)CC)cccc(SC)c1[N+](=O)[O-] c1(NC(C2C(O)CCN2Cc2ccnc(Br)c2)=O)nc2cc(Cl)ccc2s1 c1(OCC)nc(N2CC3CC2C3OC)cc(C)n1 N1(C(c2c(C)[nH]cc2)=O)CCC(C(F)F)(CNC(c2c[nH]cc2C(F)(F)F)=O)C1 c1(C(N2CC(F)(CNC(=O)Cc3ccsc3)C2)=O)c[nH]c2cc([N+](=O)[O-])ccc12 c1(N(C)CC2CCN(C(c3ccoc3)=O)C2)ncnc2cnccc12 Cc1c(F)ccc(Cl)c1C(N1CCCC(CO)(NC(=O)C(O)CC(C)(C)C)C1)=O N1(C(CCn2cc(CCCNCCCCC)nn2)=O)CCN(CC(C)(C)O)CC1 C1(C(=O)NCC(C(C)(C)C)NC(C2(C3CC3)CCC2)=O)CC2(C1)CC(F)(F)C2 C1(CNC(=O)C(F)Oc2ccc(F)cc2)CCC2(CCNC2=O)CC1 C(=O)(C1=NOC(C)C1)NC(C1(CNC(c2ccnc(C)n2)=O)CC1)C N1(c2ccnc(SC)n2)CC2CCC1CN2C(c1c(I)ccnc1Cl)=O C1(O)(CC(=O)N(CCCN(C(c2cccc(C)c2)=O)C)C)COC(C)(C)C1 CN1CCCCC1C(=O)NCC1CC(O)(CNC(=O)C(F)CC2CCCCC2)C1 N1(C(CC(C)C2CCCCC2)=O)CCCC(NC(c2cc(O)ncn2)=O)C1 C1(OCC(=O)NC(CCOC)CNC(=O)C(n2nccc2C)C)CCC(C)CC1 C(c1ccccc1Cl)=C(C)C(N1CC(NC(C2CC3(CCC3)C2)=O)C(O)C1)=O C1(C(=O)NC(C2(O)CN(C(=O)CCc3nccn3C)C2)C)CC2(C1)CC2F c1(OC)nc(C)ccc1C(N1CC(NC(=O)Cn2ccc(=N)[nH]2)C(C)(C)C1)=O c1(C(C(=O)NC2CN(C(=O)CC3CCSC3)C2)N(C)C)ccc2ccccc2c1 CN1CCCC12CN(C(C1CCCC1NC(=O)Cn1cccnc1=O)=O)C2 C1(C(N2CCCC(CCNC(c3cnc(C4CC4)o3)=O)C2)=O)CC2CC(=O)C1O2 N1(C(CCCC(CC)NC(=O)CCCCC(N)=O)=O)CCC(C2CCCC2)C1 Cc1noc(C(C)NC(C2CCC(NC(C3COCC3C(N)=O)=O)C2)=O)n1 C1(NC(c2c[nH]nc2[N+](=O)[O-])=O)CCOC2(CCN(C(C34CC3C4)=O)CC2)C1 Cc1cc(C)c2c(c1)N(C(c1nnn(C)c1C)=O)CCC2 C1(CNC(=O)COC(F)(F)F)CN(C(C2CCCS2)=O)CCC12CCOCC2 c1(C(C)=O)c(C)[nH]c(C(N2CCC(CNC(=O)C3CC3)C2(C)C)=O)c1C(C)C n1(CC)c(O)nc(OC(=O)C(CCCOC)NC(=O)OC(C)(C)C)cc1=O N(C(=NCC1CCN1C1CC1)NCC1(O)CCCC1)C(C=C)C N1(C(CC2CC(CC)C2)=O)CCC(CNC(c2cccc(C(F)F)n2)=O)C(C)C1 c1(CNC(C2N(CC)CC2)=O)cccc(CO)c1.c12ccc(o1)C(=O)NCC2 c1(CNC(=O)NCCOC2CCS(=O)(=O)C2)ccc(O)c(Br)c1 N1(C(CC2CCC(=O)NC2)=O)CCCC2CN(C(C3(C(F)F)CC3)=O)CCC12 C1(C(N2CCN(C(C3CC(O)C3)=O)C(C(C)C)C2)=O)(OC)CCS(=O)(=O)C1 C1(N(C(=O)CCC2CCCCC2)CC)CCCN(C(c2c[nH]ccc2=O)=O)C1 c1(CNC(N(C(C)CO)C)=O)ccc(Br)c(N)n1 n1(CC(=O)NCC2CCCC(NC(CCSCC)=O)C2)ncn2nccc2c1=O c1(C(N2CCC(O)C2(C)C)C(=O)N(CC)CC2CCCCC2)ccc(Br)c(Cl)c1 c1(-c2cn(CCC=C)nn2)cnn2c1CN(C(c1cnc3[nH]nnc3c1)=O)CC2 c1(C(N(CC(C)NC(c2cnc(O)n2C)=O)CC)=O)cc(C)c2n[nH]cc2c1 C(N=c1[nH]c(Cl)nc2c1CCC2)C1CC(C)N(C(=O)C=Cc2ccncc2)C1 CCC(C)C(C)C(=O)NC(C)C(CO)NC(=O)C(F)C(C)C Cc1ccc(F)c(C(N2CC3CN(C(=O)CC4CCC(C)C4)CC(C2)O3)=O)c1O c1(C(=O)NC(C=C)C(=O)NC)ccc(CNCC2CCCC(C)C2)cc1 CCC(C#N)(CC)C(=O)N1CCN(C(C2CC2Br)=O)C(C)C1 Cn1nc(I)cc1C(=O)OC(F)(F)C(F)Cl N1(C(Cc2c(C)n[nH]c2C)=O)CC2(C1)C(NC(C13CCC(C1)C3)=O)CCS2(=O)=O c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CCCCCC1NC(=O)CCC(N)=O c1(C(c2n(CC(=C)C)nnn2)NCCc2noc(CC)n2)ccc(C)cc1 c1(CC(N2C(C(=O)Nc3cc(C(=O)OCC)[nH]c3)CC2)=O)ccccc1[N+](=O)[O-] N1(C(c2cc(C)ncc2)=O)CC(C)(C)OCC1CNC(=O)COCP(C)(C)=O C(C)(CCC(=O)N1CCCC1CN(C(=O)Cc1c[nH]nc1C)C)N(C)CC CC(C(=O)N(C)CCN(C(C1CCCCCC1)=O)C(C)C)C(C)S(C)(=O)=O C(=O)(CC(F)(F)C(F)(F)F)NC(C(CO)NC(CCn1ncc(C)c1)=O)C N1(C(C23CC(n4cc(-c5ccc(C)cc5)nn4)C2C3)=O)CCC2(CC1)CC2C#N C1(C(=O)NC2CCC(CN(C(=O)CC(F)(F)F)C)CC2)CC2CCC(C1)O2 CN=c1[nH]ccc(C(=O)NCC=CCNC(C2(F)CCOC2)=O)c1[N+](=O)[O-] C(=O)(CS(=O)(=O)CC1CCCO1)N1CC(OCCNC(C2(C)CCC(=O)N2)=O)C1 C(C1c2ccsc2CCN1C(=O)CC1CC=CCN1C)NC(CC(C=C)(C)C)=O c1(CN2C(C(N(C(C)CNC)CC)=O)CC2)cc(-c2ccncc2)no1 C1(C)(C(=O)NC2C(CNC(CCCC=C)=O)C2)CC(C2CC2)=NO1 S1(=O)(=O)c2ccc(c(Br)c2)NCC2CCN2N1.C=CC1(OC)CCOCC1 C12(NC(C3C(CC)CCO3)=O)CC1CN(C(c1cnn(C(C)C)c1Cl)=O)C2 CC1CN(Cc2cccc(Cl)c2)CC(C)N(C(=O)Cc2ccon2)C1 C(=O)(C1CCc2cc(Cl)ccc21)NCC(CNC(C1N(C(C)C)CCC1)=O)O c1(OC)cc(C(N2CCC(O)(C(C)NC(c3cc(C)no3)=O)C2)=O)cc(C)n1 C(C(F)(F)CCC(=O)NCC(C)(O)CC(C)C)n1cc(C2(COC)COC2)nn1 c1(C(C)O)nc(COCC(F)(F)C(F)F)n(-c2ccc(C)cc2)n1 Cc1ccccc1COCCC(N1CCC(NC(C2(C#N)CCCO2)=O)C1)=O C1(C(=O)NCC2C(C)(C)CN(C(C3CC3C#N)=O)C2)CCC2(CC1)CC(O)C2 c1(C(=O)NCCC2CC(NC(c3ccc(Cl)s3)=O)C2)cnc(O)c2cncn12 c1(C(=O)NC2CC(NC(c3cccc(O)c3Br)=O)C2)ccc2ccnn2c1 c1(C(=O)NCC2CCC(F)(CNC(CC(COC)C)=O)C2)ccc(Cl)nc1OC O=C(C1=CCN(C(=O)CC23CCCC2C3)CC1)NCCc1cncnc1O C1(CC=C)(NC(=O)CC2CC2(Cl)Cl)CCN(C(=O)C=Cc2ccncc2)C1 Cc1nccn1C(C)C(=O)NCCCN(C(c1c[nH]nc1OCC(C)C)=O)C(C)C c1(OCC(=O)NC(CN(C(=O)Cc2cccs2)C)CO)ccccc1.C(CF)O c1(C(=O)OC)ccc(C(=O)NCC2CCN2C(=O)C(O)C(F)F)cc1Cl C1(NC(COCP(C)(C)=O)=O)CC(NC(c2ncc[nH]c2=O)=O)C12CCC2 C(=O)(C1CCCc2ccccc21)N1C(C(=O)Nc2cc(Cl)ccc2O)CC(OC)C1 C1(C(N2CCC(N(c3nccs3)C)CC2)=O)CC12CCCOC2 c1(CC(=O)NCC(C2CCCC2)NC(C2(n3cnnn3)CC2)=O)cccc(F)c1F N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(c2cnn3cnnc3c2)=O)C2CCCC12 c1(C(=O)NC(C(C)C)CNC(c2ccc(C3CC3)o2)=O)ccc(=O)n(C2CC2)c1 N1(C(=O)NCC(=O)NCC#C)CCC2CCOCC2C1 CCC(CC)C(C)C(=O)N1CCC2CCCC12CNC(c1ccc(OC)cn1)=O C(N=c1[nH]cnc(C)c1Br)C1CCN(C(c2c(CC)cccn2)=O)C1 C1(C(=O)NCc2ccc(C(=O)NCc3n(C)nnn3)o2)C2CC3C(C2=O)C13 Cc1cc(C)c(CC(N2CCCC(CNC(=O)CN(c3ccncc3)C)C2)=O)s1 Cc1ccc(CC(=O)NCC2CN(c3nc(C(C)(C)C)ns3)CCN2C)c(Cl)n1 N1(C(CCC)=O)CCCC2(CCN(C(C3CC4COCC4C3)=O)C2)C1 N1(C(CNC(c2ccc(OCOC)cc2)=O)C(C)C)CC(C)OC(C)C1 C(=O)(CCCCC(=O)NCCC1(NC(C23CCCC2(C(N)=O)C3)=O)CC1)NC c1(C(=O)NC2CC(C(=O)Nc3cnc(C(F)F)cn3)C2)cc(Cl)cc(Cl)c1Cl C(=O)(CC1=NNC(=O)C1)N(CCCNC(c1cc(N)cc(O)n1)=O)C c1(C(N(C)CCOCCNC(C2CC(CCO)C2)=O)=O)cc2cccc(O)c2[nH]1 N1(C(C(CC)n2cc(-c3cnc(OC)c(C)c3)nn2)=O)CC2C(C1)C2(C)C CN=c1nc(C(N2CC(F)(F)CC2CO)=O)cc(C)[nH]1.C12CCCC1NC2=O N1(CC(=O)NC(C(C)(C)NC(c2cc(CC)no2)=O)C)C(=O)NC(C)(C)C1=O C(=O)(CCC1CC1(C)C)NCCN(C)C(=O)NC(=O)OC(C)(C)C C(=O)(CCC(=O)NN(C)C)NCC1C(CNC(c2ncc(C)cc2C)=O)C1 C(N=c1[nH]c(C)nc2c1CCCC2)C1(OC)CCOC1 C1(NC(CN2CC(CC)C2)=O)CCCC12CN(C(c1cc3n(n1)CCO3)=O)C2 N1(C(=O)NCc2ccc(C(C)C)[nH]2)CCc2ncn(C)c2C1 C1(CNC(C2CC(NC(COC3CC(C(N)=O)C3)=O)C2)=O)C=CCOC1 C1(C#N)(C(=O)NCCN(C(C(c2cnn(C)c2)OC)=O)C(C)C)CC12CCC2 c1(CC(C#N)NC(C(c2ccc(C(C)(C)C)cc2)(F)F)=O)ccccc1[N+](=O)[O-] N1(C(c2c(CC)ccs2)=O)CCCC2(CCC(NC(C3(CO)CCCC3)=O)C2)C1 c1(C(=O)NCC(CNC(CN(C)Cc2ccccc2)=O)CO)cnc2n1CCC2 c1(C(N2CCC3(C2)CN(C(C2CC2F)=O)C3)=O)cc2ccc(Br)cc2cn1 N1(C(c2c(NCC)scn2)=O)CC2(CCN(C(=O)Cc3ccccc3F)C2)C1 C1(CNC(C2(OC)CCSC2)=O)CC2(CO1)CN(C(=O)CCC1CC1(F)F)C2 O=S(=O)(c1cccnc1NCCc1cccs1)N1CCN(CC2CCC2F)CC1 CC(C)CC(Cc1ccc(F)cc1)N=c1[nH]c2c(c(=NCCF)[nH]1)COC2 Cc1ccc2sc(N3CCCC(C#N)C3)nc2c1 n1(CC)nc(C(=O)NC(C)CN(C)C(c2sc(C)cc2C)=O)cc1O C1(C(N2CC(C(=O)OCC)C2)=O)CCCN1C(=O)CCCC1CCCO1 C1(C(=O)NCCC2CCN(C(CCN(C)C)=O)C2)CCCCCC1 N1(CC(N2CC(C)(NC(=O)OC(C)(C)C)C2)=O)CCC(=O)NC1=O C(CCCCCN(C(=O)C(c1cccc(Cl)c1)(C)C)C)NC(CC(C)OC)=O CCCC(C(=O)NC1CC1NC(=O)CCCNc1nc(C)cs1)N(CC)CC C(CC(C(=O)N(C1CC(SC)C1)C)NC(c1ccccc1NC)=O)OCC c1(NCC(N2CC(C(C)NC(c3c(CC)nc(C)[nH]3)=O)C2)=O)ccc(Cl)cc1Cl N1(C(=O)CCCN2CCCC2)CCCC(CNC(c2ccc(F)cn2)=O)C1 c1(C(=O)NC(C2CN(C(C(C)SCC)=O)C2)C)cc[nH]c1C(C)C C1(C(N2CC(NC(=O)Cc3noc(C)c3C#N)C2)=O)(COC)CCC(F)(F)CC1 N1(C(C2N(C(Cc3c(CC)con3)=O)C(C(C)C)CC2)=O)CCC2(CCCC2)C1 c1(NC(C(=O)NC(C)CCN2CCCCC2)=O)cnn(-c2ccc(F)cc2)c1N Cc1nn(C)c(C)c1C(C)C(=O)NC(CNC(=O)CS(=O)(=O)NC1CC1)C(C)C C(=O)(CCCC(C)(C)C#N)N1CC(CCNC(CCCCCOCC)=O)C1 C1(C(CNC(=O)CC=C(C)C)NC(CCN(C)CC)=O)CC=CCC1 Cc1ccc(CNc2ccc(NC(c3ccnc(F)c3)=O)c(F)c2)c(F)c1 C#Cc1cc(F)ccc1CN1CCN(C(c2ccncc2Br)=O)C(CC)C1 C(=O)(CC(C)CC(=O)N1CCCOC(CNC(=O)CCCn2cccn2)C1)OC C(=O)(CCCC(F)(F)F)NCC(CN(C(CCn1c(C)csc1=O)=O)C)(C)C c1(C(N2CCC(c3nc(C)on3)C2)C(=O)NC2(C)CC2)cn(C)nc1C1CC1 CCCC(CC(=O)N1CC=CCO1)NC(c1ccc(C)c(C#N)c1)=O c1(C(=O)NC(CNC(C(F)=CCC)=O)C2CCC2)cc2c(Cl)nccc2o1 Cc1cc(OC(C)(C)C)ccc1C(F)(F)F.N1(C(=O)N)CCC(N(C)C)CC1 CC(C(=O)NCC1(F)CCC(NC(=O)CNC(=O)OC(C)(C)C)C1)C(C)(C)C c1(C(=O)NC2CN(C(=O)CCCCCF)C3(CCC3)C2)cc(F)cc2nn[nH]c12 CCC(C)(CNC(c1scnc1C)=O)C(=O)NC(CCO)C(C)(C)O Cc1ccc(C(=O)NCC2CCCN(C(=O)CCN3CCCC3)C2)c(C)c1 C#Cc1ccc(C(N2C(C(N3CCC34CN(C)C4)=O)CC2C)=O)nc1 C1(C(C)C)CCC(C)CC1C(N1CC(CF)(NC(=O)C(C)CF)C1)=O c1(-c2cn(C(c3ccc(OC)cc3)C)nn2)cccc2ncccc12 CC1CCN(CC(=O)N(C2CC2)CC2(n3cnnn3)CCSCC2)CC1 N1(C(c2c(CC)ocn2)=O)CC2CN(C(C3CC4CC4C3)=O)CC2C1 Cc1sc(C(=O)OC(c2ccc(OC(F)F)cc2)C)nc1C(F)(F)F S(=O)(=O)(c1ccc(Cl)c(C(=O)NCCCNC(C2CC2C#N)=O)c1)NC Cc1onc(CC(=O)N(CC(C)O)CCNC(C2(NC)CC(F)(F)C2)=O)c1C#N N1(C(CC2N(C(C(C)SC(C)C)=O)CCC2)=O)C2COCC1C2 C12(C(N3CC(OCC(=O)NC4CCCC45CCC5)C3)=O)CCC(CC1)CC2 c1(CCC(=O)NCC(CN(C(c2c(NC)snc2C)=O)C)C)cc(C)cc(C)c1 c1(CC)ccc(C(=O)NC2CCCC2NC(=O)CC(C)n2ccnc2)s1 c1(C(OC)OCC)ccc(CNC(C2CC3CCC2C3)=O)c(F)c1 C#Cc1c[nH]nc1C(=O)NC(C1CCCCC1)CNC(C1(Cl)CC1(F)F)=O N1(C(C(C)NC(C)=O)=O)CC(C)(C)OCC1CNC(c1cccc(N)c1)=O Cc1nnn(CC(=O)NC(C)CN(C)C(C2CCCSS2)=O)n1 C1(C(=O)NCC(C)(C)C2CCC2)CC(NC(=O)CC2CC3C=CC2C3)C(O)C1 N1(C(COC(CC)CC)=O)CCCC(C)(C(=O)NC2CC(CSC)C2)C1 C(=O)(C1(C)OCCc2ccccc21)NCCC1N(C(C=CCC)=O)CCCC1 C=CCC(C)C(=O)N(CC)CC1CCN(C(=O)CCCOC(C)(C)C)CC1 CC(C)C#CC(=O)NCCCOCCN(C(=O)CC(C)Cc1cccc(F)c1)C C1(C2CCN(C(C3CCN4CCOCC34)=O)CC2)(NC(C(C)S(C)(=O)=O)=O)CC1 C1(NC(c2sc(C)c(O)n2)=O)C(C)CCN(C(c2csc(Cl)c2)=O)C1C C12(C(=O)NC3C(NC(c4c(OC)nsc4)=O)COC3)CCC(C1)OC2C N1(C(CCCC#C)=O)CC2CC3CC2C1C3NC(C1CC2CCC(C1)C2O)=O C1(NC(C2CCC(=O)N2)=O)C2CC1N(C(C13CCC(CC1)O3)=O)C2 c1(SC)cccc(C)c1C(N1CCCC(c2nccn2C)C1)=O C1(OC)CC(NC(C2CC(C(C)C)C2)=O)CN(C(c2cocc2C)=O)C1 C(=O)(C1COc2ccccc21)NC(C(C)C)CCNC(=O)CC1CC2CCC1O2 N1(C(C=C(CC)C)=O)CC2CCCC2(NC(=O)C(O)CC2CCCCC2)C1 N1(C(=O)NC2CC3COC2C3)CCCCCCCCCC1 c1(OC)cnc(Br)cc1NC(C1CC12CN(C(=O)CCN1CCOCC1)C2)=O c1(CCC(N2CC(C)N(C(C3CC4(CCC4)C3)=O)CC2)=O)ccc2c(c1)CCO2 C1(C(=O)NCC2CC(NC(c3cnn(CC4CCCO4)c3)=O)C2)CCC2(CC2)C1 c1(SCCN(C(C2(C)CCCO2)=O)CC)ccccn1.C(=O)C(C1CCCO1)C1CC1 c1(C(=O)NCC2(Nc3c(C)cnc(Cl)n3)CCCC2)ccc2[nH]ccc2c1 c1(C(=O)NCC2(CC)CCCO2)coc2c1CN(C(=O)CN=[N+]=[N-])C2 c1(C(=O)NCC2CC(NC(C(CC)NC(N)=O)=O)C2)ccc(C)c(Br)c1F C(CNC(=O)Cn1cnnn1)(C(=O)NCc1nc(CO)n[nH]1)N(C)C CC1CN(C(=O)CC(C(C)(C)C)NC(c2ccco2)=O)CC(C)(C)CO1 CCCC(C)CCCC(=O)N(C1CCN(C(=O)CSc2nccn2C)C1)CCC C12CCC(CC1)C(=O)NC2.C1(F)(C(=O)NC2CC(C(C)(C)C)C2)CCCC1 N1(C(C(=Cc2n(C)ccc2)F)=O)CCN(C(C2C(F)(F)C23CC3)=O)C(CO)C1 CC(CS(C)(=O)=O)C(=O)N1CC2(CNC(=O)CN(c3ccccc3)C)CCC1C2 Cc1c(Br)c(C(=O)NC2CN(C(c3cnccc3Cl)=O)CC2O)nn1C Cc1cccc2[nH]c(CN3CCCC(n4cc(C(=O)O)nn4)C3)cc12 CCCCCCC(CC)C(=O)N(CC(C)NC(C1CC1c1cnn(C)c1)=O)C C(=O)(C(C)(C)CCCNC(=O)CCCCC(C)C)NCC(C)OCC=C CCCCC(O)C(=O)N1CC2CC1CC2CNC(c1ccc(CC)cc1N)=O c1(CN(C(C(N)C(F)(F)F)=O)CC(=O)O)nc2c(s1)CCCC2 CC1=NOC2(CCN(c3ncccc3S(=O)(=O)NCCc3cc(C)no3)CC2)C1 C1(C2CC2)(C(=O)NCc2ccc(C(=O)NCCP(OC)(C)=O)o2)CC(=O)C1 Cc1cc(F)c(C(N2CC(C3CN(C(c4ccnc(C)c4)=O)C3)C2)=O)c(Br)c1 C=CCC(CC(=O)N(C)CC1CCCCC1)NC(C1(C)CCC2CC2C1)=O N1(C(CCCC)C)CCC(C(=O)NCC(C)CC(=O)N2CCOCC2)CC1 O=S(=O)(c1ccc(NC(Cn2ccnc2)C2CC2)c(F)c1)NCC=CBr C#CCC(CC#C)C(=O)NCCN(C(=O)C(C)C1CC1)CC1CC1 c1(C(=O)NC(CCN(C(C(CC)c2cccnc2)=O)C)(C)C)cccc(Cl)c1 CC1CN(C(=O)CC2CCCCN2C)CCN(C(c2ccc(C(C)(C)C)s2)=O)C1 C#Cc1cccc(C(=O)NC(CNC(=O)CC2CCC(C)CC2)CC)c1F c1(CC)nc(C)ncc1C(=O)NCCC1CCC(NC(=O)C2CC2)C1 N1(C(=O)NC(C(C)C)c2ccco2)CCC(Cc2ccoc2)CC1 c1(COC)cccc(NC(=O)C(=O)N(CCN(C)C)CC2C=CCC2)c1 CC1CN(C(c2ccc(C3CCC3)nc2)=O)CCC1CNC(=O)CSC(=N)N CCC(C(=O)NC(COC)C(=O)NCCF)C(C)(C)CC Cc1cc(O)ccc1CNC(=O)CC1CSC1.C12(CCCC1)CCC(=O)N2 Cc1nc(=N)[nH]cc1C(=O)NCC1COCC1NC(=O)CC1(O)CCCOC1 C(c1cn[nH]c1)=C(C)C(=O)NC(Cc1cnc[nH]1)C(=O)NCCCCCF c1(C2CC(C(C)C)O2)nc(-c2cscn2)nn1-c1ccnc(Cl)c1 C#Cc1cnc(C(N2CC3(CC3)CC2CC(=O)N(C)Cc2ccsc2)=O)c(C)c1 c1(OC(C)C(=O)NCC2CC2CC(=O)NCCC)n[nH]c(C2CC2)c1C.C1CO1 CC1CN(CCCC(c2ccc(Cl)cc2)=O)CC(c2ccc(F)cc2)O1 O=C1CC2CC1NC2NC(c1ccc(CC(F)F)cc1)=O C1(NC(c2ccc(CCC#C)cc2)=O)CCCCN(C(=O)C(C)NC(=O)NC)C1 C1(C)(CC)C=C(C(=O)NCC2CC(OC)CN2C(c2ccc(O)cc2)=O)C1 c1(C(N2CCC(N(C(CCCSC)=O)C)C(C)C2)=O)ccn2[nH]c(=N)nc2c1 CC(N=c1cc[nH]cc1S(=O)(=O)NCCCN(C)C)C(C)c1ccccc1 C(N=c1cc[nH]cc1S(=O)(=O)NCCCCN(C)C)c1nnc(C)s1 N1(C(C(C)CN(C)C)=O)CCCCC2(C1)CN(C(=O)C1CCCc3ccnn31)C2 C(CCN=c1[nH]c(=NCC2CC(O)C2)[nH]c2cc(OC)ccc12)N(CC)CC C12(OC)CCCC(C(=O)Nc3cnccc3C(c3ccc(F)cc3)=O)(CC1)C2 C1(C(=O)NCC(C)(C)NC(C2(CC=C)CC2)=O)CCC(=O)N1CCC C#Cc1ccc(CN2CC(O)CC2C(C)C)c(Br)c1 N1(C(c2ccc(C(C)C)cc2)C)CC2CCC(NC(=O)CC(C)C(C)C)CC2C1 C(C(CC(F)(F)F)NC(=O)Cc1c(Cl)cnn1C)NC(C1N(CC)C(=O)CC1)=O C1(CC(=O)NC)CCCN1C(=O)C=CC(C)NC(C1CCCN1C)=O C1(NC(c2ccc(F)nc2)=O)CN(C(c2cnoc2)=O)CCC12CCC2 c1(CC)cc(C(=O)NC(C)C(C)NC(=O)CCn2cncn2)ccc1Cl C(=O)(CCCS(N)(=O)=O)N1CC2C(NC(C(CC)NC(C)=O)=O)C2C1 C1(NC(c2cc(C)oc2C)=O)CN(C(=O)CN2CC(=O)N(C)C2=O)CC1(C)C c1(OC(C(=O)N(C)Cc2ccc(Cl)cc2)(F)F)ccc(Cl)c(Cl)c1 CCC(CC(=O)N1CC(CNC(c2cncs2)=O)CC1(C)C)C(F)F Cc1cccc(C(=O)NCC2(C)CCN(C(=O)C=CC3CCOC3)C2)c1C C(=O)(C#CC1CCOC1)N(CCCCN(C)C(c1ccnn1C)=O)C C1(CNC(C(CC2CCOCC2)NC(c2c(C)nco2)=O)=O)CCCC(=O)N1 C1(C(N(C(CC(=O)NC2(CSC)CCC2)(C)C)C)=O)C2CCC(F)C12 CC(C)(C)CCC(=O)N1CCC1C(=O)NC1(C)CCN(C(=O)OC(C)(C)C)C1 C12(C(=O)NCC3N(C(C4(C)CC(C)(C)C4)=O)CCCC3)CCC(C)(CO1)C2 C(CCCCCN(C)C(C1(C)C=CCC1)=O)NC(c1ccc(C(C)=O)o1)=O N1(C(c2c(OC(F)F)cc(C)s2)=O)CCC(C)C(CNc2cc(=O)n(C)cn2)C1 n1(CC)cnc(CCNC(=O)N(C(COC(C)C)C(=O)OC)C)c1 C1(C(N2CC(CCCCNC(=O)COC3CCCOC3)C2)=O)CC12CC(O)C2.CCC C1(CNC(C(C)(Cl)Cl)=O)CCC(NC(=O)C=CC2CCCCC2)CC1 c1(N(CCN(C(c2cc(SC)oc2)=O)C)C)nc2cc(C)ccc2o1 CC1(C(N2CC=C(CNC(C3CC4C=CC3O4)=O)CC2)=O)CCCCNC1=O S(=O)(=O)(c1cc(C(N2CC3C(NC(c4cnc(Cl)[nH]4)=O)C3C2)=O)co1)N(C)C c1(CN)ncc(C(=O)NOC2CC(F)(F)C2)o1.C1(C(C)C(=O)OC(N)=O)CCNC1 C(C(C)(C)CNC(=O)C(C)NS(=O)(=O)CC)N(C(=O)CCn1ccc(C)n1)CC c12cc(ncn1)NCCN2CCC.N1(Cc2ccc[nH]2)CCOCC1 N1(C(CC=C)=O)CC(CNc2nnc(C)c(C)n2)CC(C)(C)C1 c1(CC(C#C)ON)c(C)nsc1-c1ccnn1C C1(C(=O)NCC2CCCOC2)CC(F)CN1C(c1n[nH]cc1Cl)=O Cc1cnc(CN(CCC(C)C)C=O)cc1C C(=O)(C(C)N=c1cc[nH]cc1)N1CCC(Cc2cn(CCOC)nn2)C1 C1(CC(=O)NC2C(NC(CC3CN(C)C3)=O)CCC2)CC(C)(C)OC1=O c1(C(=O)NC(CN(C(C(C(=O)OC)C)=O)C)C)c[nH]c2nccc(Cl)c12 C(=O)(C1=CCCCO1)N(C1CCC(NC(C2(CO)CCOCC2)=O)CC1)C C1(F)(C(=O)NCCCCCN(C(c2n(OC)cnc2C)=O)C)CC12CCCCC2 Cc1cc(C(N2CC3(CC3)CC2C(=O)NC(C2CCC2)C)=O)cc(F)c1 c1(C(=O)NCC(C)(C)OCCNC(C2(C)C=CCC2)=O)cc(Cl)cn1C C1(CNC(C2=NOC(C)(C)C2)=O)CN(C(=O)CNC=O)C2(CCOCC2)C1 N1(C(CC2(N(C(CCOCC(C)C)=O)C)CC2)=O)CCC(O)(CO)CC1 C(C(CCCC)NC(C1(n2cccn2)CC1)=O)NC(c1ccc(CCC)[nH]1)=O C1(CNC(=O)C(c2cccnc2)O)CC(F)CN1C(=O)COc1ccc(F)nc1 c1(NC(C2N(C(C(C)(C)C)=O)CSC2)=O)cc(Cl)ncc1Br O=C(CCCCc1cnc[nH]1)N1CCN(C(C2(CC(F)F)CCC2)=O)CC1 N1(C(COC(CC)C)=O)CCSCC1C(N1CCC(C)(C(=O)OC)C1)=O N1(C(C=CCCC)=O)CCC(C(=O)Nc2cccc(-c3ncon3)c2)C1CC C1(NC(c2cc(C)nn2C)=O)CN(C(c2cncc(C(C)(C)C)c2)=O)CC1(C)C N1(C(CN(C(=O)C(C)Cc2cnn(C)c2)CC=C)=O)CCc2sccc2C1 N1(C(C2CN(C(COC(C)C)=O)CC(C)(C)C2)=O)CCn2c(O)nnc2C1 CC1(C(=O)NCC#CCNC(c2ncoc2-c2cccs2)=O)CCCC1 N1(CC(=O)NCCCC)CC2(CN(C(C3CC(C)=NO3)=O)CC(C)(C)O2)C1 C(=O)(CS(=O)C(F)(F)F)NC(C)CC1CN(C(c2cncc3c[nH]nc23)=O)C1 n1(CC)nnc(C)c1C(=O)NC(C1CCN(C(C2CCC(C)(C)C2)=O)CC1)C C(C(CC(C)(C)C)OC)N(C(c1ccccc1)C(=O)NCC=C)C C1(COC)CN(C(c2ccc(F)c(Cl)c2)=O)CCN1C(=O)C#CC(C)(C)C N(C1COc2ncc(C(F)F)cc21)C(=O)Nc1cccc(Oc2cccnc2)c1 CCC(C)C=CC(=O)NCC1CCN1C(c1ccc[nH]1)=O c1(CC)ccccc1C(CNC(c1ncoc1C1CC1)=O)NC(=O)CCC#N CCCC(C(=O)N1CCCC(C(=O)NCc2ccncc2F)C1CC)OC c1(CC(=O)NC(CCCNC(Cc2scc(CC)n2)=O)C)c(C)cc(C)cc1C C1(NC(C(C)(C)C(N)=O)=O)CN(C(=O)C2=CCCOC2)CC2(CCC2)C1 C1(CC(=O)N(CC(N2CCCC2)C)C)(NC(C2CCC2(C)C)=O)CCOCC1 c1(C(=O)NCC2CC(NC(CCCCC#C)=O)C2)cc2ccccc2nc1OC C1(NC(CCCC(=C)C)=O)CC1C1CCCN(C(=O)CCC2CCCN2C)C1 C(=O)(C1=CN=C2N=CNN2C1)NC1(CNC(c2cnc(COC)s2)=O)CC1 c1(CNC(=O)C(=O)NC2CC(=O)NC2=O)ccc(CC2C3CCOCC23)cc1 Cc1nn(C)cc1-c1cn(CCOCCNC(=O)Cc2nn(C)cc2Br)nn1 CCC(CC)C(F)C(=O)NCCC1CC(C(=O)NCC(c2ccccn2)C)C1 N1(C(c2ccc(C)nc2O)=O)CC(C(=O)NCC2CC23CC3)CC(C)(C)C1 N1(C(CCC#CC)=O)CCN2CCN(C(=O)C(CC(C)C)NC(C)=O)CC2C1 C1(N(C(c2c(OC)ccc(O)c2)=O)C)CCN(C(c2cn(C)nn2)=O)CC12CC2 CC(C)(C)C(O)C(=O)N1CCCC1CC(=O)NCCCC1(O)CCC1 N1(C(CC(C)(C)N(C(C2CN(OC)C(=O)C2)=O)C)=O)CC(C)C12CCOCC2 C(=O)(C(C)(C)C(C)(F)F)NCC(CNC(CCOC)=O)C(F)(F)F C(C(COC)C(=O)N(CCCN(C(C)=O)CCOCC(F)(F)F)C)OC c1(C(=O)NC(C)CCCNC(=O)CCCS(N)(=O)=O)ccc2c(c1)OC(C)(C)O2 C1(NC(c2n(CC#C)ccc2)=O)CN(C(=O)C(C)CC(N)=O)C2(CCCCC2)C1 c1(-c2n(CC3CCN(CCOC)CC3)c(N(C)C)nn2)cc(F)c(F)c(F)c1 c1(CC)cncc(C(=O)N(C2CC(NC(=O)CCOc3cccc(F)c3)C2)C)c1 Cc1cc(F)ncc1C1CC(CNCCC2CN(C(C3CCC(=O)C(C)C3)=O)C2)C1 C1(CNC2CCCCN(C(CSCC)=O)C2)CC12CCC(F)(F)CC2 C1(CNC(c2cc(CC)no2)=O)CC(F)CN1C(c1cnn(C2CC2)c1C)=O N1(C(C2N(S(C)(=O)=O)CCCC2)=O)CCCCC(CNC(c2cnco2)=O)C1 C=C(C)CC(C)C(=O)N1CCCOC(Cc2ccccc2)C1 C1(n2c(C(=O)OCC)ccn2)CN(N2CCCC2CC(N)=O)C1 O=C(C1=CCC(F)(F)CC1)NCCC1(O)CN(C(c2cn3c(n2)CCCC3)=O)C1 Cn1ccc2c(C(N3CC4CC3C4NC(=O)C(C)(C)C3CCC3)=O)ncnc12 CC1CN(C(=O)C(=O)C(C)(C)C)CCC1NC(=O)CC1CCCC(C2CC2)O1 C1(CC=C)(C(=O)NC2CCC2NC(=O)CNC(c2ccco2)=O)CCC1 C1(CNC(CN2CCCC(CC)C2)=O)CN(C(=O)C#CC2CCC2)C(C)(C)C1 CC(O)(CNC(=O)CC1CC12CC2)CNC(C1(C(=O)OC(C)(C)C)CCC1)=O C(=O)(C(C)(C)CC(=O)OCC)OCCc1ccc(C(=O)Nc2nnco2)cc1 c1(C(=O)NC2CN(C(C(COC)(C)OC)=O)CC2C)cnc(C)[nH]c1=N n1(CCC)nnnc1C(c1ocnc1CC)NCCc1nccn1CC C1(NC(C(CC=CC)C)=O)CC2CCC(C1)N2C(c1cnc(OC)nc1)=O c1(C(=O)NC(CC(C)NC(c2n[nH]c(=N)[nH]2)=O)C)ccc(-c2ccncc2)cc1 c1(CC(=O)NC2CC(NC(C(C)NC(CC)(C)C)=O)C2)ccc2c[nH]nc2c1 C(C(O)CCNC(=O)Cc1cc(C)ns1)NC(CC1(OCC)CCC1)=O CC(C)(C)CCC(CO)NC(C(=O)NCC(c1cccc(Br)c1)O)=O c1(CC(=O)NC(C)CCCNC(C2(F)CC2)=O)ccc(-n2ccnc2)cc1 c1(NC(C2C(C)(C)C(NC(c3c[nH]c(C(N)=O)c3)=O)C2)=O)ccc(Cl)c(O)c1 c1(C(N(CC(C)NC(c2ccnn2C(F)F)=O)C)=O)cc2n(n1)CCOC2 Cc1nc2ncccc2cc1C(=O)NCC=C1CCN(C(c2cn[nH]c2)=O)CC1 c1(OC(C)C(=O)OCC(C)(O)C(F)F)cccnc1N(C)C C1(N(C(c2c(OCC)ccs2)=O)C)CCN(C(=O)CCCF)CC1 C1(NC(c2ccc(OC)s2)=O)CC2CCC1CN(C(=O)CC1CCC(C#N)C1)C2 Cc1ncsc1C(=O)NCC(=O)NC1CCC1NC(c1cscc1Cl)=O n1(CC)nnc(C(=O)NCC2C3CC2N(C(C2COC(=O)N2C)=O)C3)c1C Cc1ccnc2sc(C(N3CCCN(C(=O)COC(C)(C)C)C(C)C3)=O)c(C)c12 c1(C(=O)NCC(CC=C)NC(C2CCCN(C)C2)=O)cc(C2CC2)cc(F)c1 c1(C(=O)NC2CN(C(CN(CC)CC)=O)CC(O)C2)cc(F)cc2nn(C)cc12 N1(C(c2c(C)cc(C)o2)=O)CC2CN(C(C3(C)CCOC3)=O)CC2(C)C1 c1(SC(CC)C(=O)NC2CCCC(NC(=O)C(O)CF)C2)ccccc1C C1(C(N(CC(C)(C)CNC(=O)Cn2ccc(Br)n2)C)=O)CCC2CC2CC1 CN1CC2CCN(C(c3ccn(CCNC(C4C=CCS4)=O)c3)=O)C2C1 C1(C(=O)NC2CC(CF)C2)CCCN1c1ncccn1 CC1CN(C(=O)Cc2csc(S)n2)CC(C)CN1C(=O)CN1C(=O)CCCC1=O c1(C(=O)NC(C)CCCNC(=O)C(c2ccccc2F)(C)F)ccc(Cl)nc1N c1(OC)ccc(Cl)c(CC(=O)NC2CCCC2NC(c2occc2C(C)C)=O)c1 C1(N(C(c2c(CC)cc[nH]2)=O)C)CCCC(NC(=O)Cn2ccc(C)n2)C1 N1(CCC(N2CC(C(C)NC(C=CC(C)C)=O)C2)=O)CCCC1=O c1(-c2cc(C(N3CCC(OCCN(CCCO)C)C3)=O)sn2)ccc(Cl)cc1 C(=O)(C1CCCc2ncnn21)N1CC(CCCCNC(CC(C)(C)C)=O)C1 CCC(C)CN=c1[nH]c(C(=O)N=c2ccn(-c3ccccc3C#N)[nH]2)cs1 C1(N(C(C2=C(C)OCCS2)=O)C)CCCC2CN(C(=O)CC3CN(C)C3)CC12 c1(NC)cnc(C(=O)NCCN(CC(C)O)C(c2ccc(C(N)=O)s2)=O)cn1 CCCC(C(O)C(=O)NC(C)CCN1CCCC1)NC(C1(C)CC(F)(F)C1)=O c1(C(=O)NC2CCCC(NC(c3ccc(CO)nc3)=O)C2)cccc2nccn12 C1(CCNC(C(C)SCC)=O)COCCN(C(c2cc(CC)cs2)=O)C1 C(=O)(N(OC)C1CCOC1)c1cncc(CNC(c2c(NC)cncc2)=O)c1 C=CC1(CC(=O)NCC(C)CCC)CN(C(c2ccc(OC)o2)=O)C1 C12(NC(c3c(OCC)oc(C)n3)=O)CCC(CNC(=O)CC3(C)CC3)(C1)OC2 CS(=O)c1ccc(CC(N2CCC3(C2)CN(C(=O)C2=CCCS2)C3)=O)cc1 C(=O)(N(CCC(=O)NCC1CC(C)CO1)OC)c1cc(CC)ncn1 c1(C(=O)NCC2(C)CCN(C(c3cccs3)=O)C2)c(C2CC2)nc2sccn12 C1(C(=O)NC(CNC(c2cn(CCC)nc2)=O)C)Cc2ccccc2N1C N1(C(C2(C)ON=C(C)C2)=O)CCN2CCN(C(=O)Cc3cn(C)nc3C)CC2C1 C(CC(C)C)(C(=O)N1CCC(C(=O)OC)C1)N(C(c1nc(CCC)oc1)=O)C CCC(C)C(C)(O)CNC(C1CC(NC(=O)C=Cc2cnccn2)CCO1)=O N1(C(=O)NCC2(N(C)C(=O)OC(C)(C)C)CCC2)CC2CC(C1)C2(C)C c1(C(=O)OCC)coc2c1CN(C(=O)NC1CC(C)C1(C)C)C2 [N-]=[N+]=NC1CCC(C(N2CC(CNC(=O)CCCn3cccn3)C2)=O)CC1 c1(C(N2CCCC(NC(c3c[nH]cc(F)c3=O)=O)CC2)=O)cccc2ccoc12 C1(C(N(C)CC2N(C(C(C3CCOCC3)OC)=O)CCC2)=O)CCOC(C)(C)C1 CC(C)(CCCNC(c1cccnc1O)=O)C(=O)NC(CC1CCCC1)CO N1(C(C2CCCN(C(CC)=O)C2)=O)CC2CCC1CN2C(c1ccnn1C)=O c1(C(N(CCC)CCCCOCC(=O)N)=O)nc(OCC)cc(O)n1.OC C1(C(C)NC(C2COCCO2)=O)(C(=O)NC2CC(OCC(N)=O)C2)CC12CCC2 CC1CC(CNC(=O)Cc2nc[nH]n2)CN1C(=O)CC1CC2(CCC2)C1 N1(C(c2cc(CNC(=O)CC3CSC3)no2)=O)C2CCC1CC(CO)C2 CN1C(=O)CCCC1C(=O)NCC1COCCN1C(c1cocn1)=O Cc1c[nH]c2ncc(C(=O)NC(C)(CNc3cc(O)ncn3)CC(C)C)cc12 CC1CCCCC1NC(=O)COCCCOCCNC(C1(C)CS(=O)(=O)C1)=O c1(CNC(=O)NCCC2C=CCCC2)nc2ccccc2[nH]1 Cn1nc(C(=O)NCC=CC(=O)NCCC2(O)CCC2)cc1F C#CC(C)(C)C(=O)NCCNC(C1CC(=O)N(CC2CC2)C1)=O CCCC(C(O)C(=O)NCCCc1cccnc1)NC(=O)CC(C)CCC N1(C(C2C(C#N)C2)=O)CC2C(CNC(=O)Cc3ccnn3CO)C2C1 c1(CCNC(=O)Nc2nn(C)nc2Br)ccc(F)c(Br)c1 CCC(O)C(C)(C)C(=O)NC1CC2CC1CN2C(=O)CCOC C(N=c1cc(C)nc(N2CCCC3(CO)CC3C2)[nH]1)c1cc(OCC)cc(C)c1 C(=O)(CCC1CC(NC(=O)COc2ccsc2)C1)N(CC(C)SC)C C1(NC(CCCSC)=O)CC2CC(NC(=O)CSc3nnnn3C3CC3)CC12 C1(CC(=O)NCC(CCC)NC(c2ccc(C)c(CC)c2)=O)CCCC(F)(F)C1 c1(OC)ccc(C(N2CCC(C(=O)NCC3(O)CC(CO)C3)C2C(C)C)=O)nc1 C1(C(N2CCC2(C)CCO)=O)(OC)CCN(C(C2CC(=O)C2(C)C)=O)C1 CC1=CCC(C(C)CC(=O)OC(c2ccc(C(=O)ON)o2)C)CC1 c1(CN2CC(C)C(CN)C2)cc(Cl)cc(Br)c1O CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)C(C)n2cnnn2)CC1C C1(CCNC(C2CC2[N+](=O)[O-])=O)CCCN(C(=O)CCc2ccccc2)C1 c1(C(N(CC(C)NC(=O)CCc2n[nH]c(=N)s2)C)=O)cc(-c2ccccc2)no1 Cc1cc(NC(c2cc(CNC(C3CCS(=O)CC3)=O)nn2C)=O)c(C)c(C)c1 c1(OC)ccc(C(N2CCC(NC(c3csc(C)c3)=O)C(F)C2)=O)c(OC)n1 CN=C(NCCCSC(C)C)NCc1ccc(C2CC2C)o1 CCCCCC(O)CC(=O)NCCC(C)NC(c1cnc(OC)cc1C(F)F)=O c1(C(=O)NC)ccc(Cn2cc(C3(NC(C)=O)CCOC3)nn2)cc1.C1C(=O)N1 c1(C(c2n(CCC)nnn2)NCc2nc(C)co2)ccc(C#N)cc1OC N1(C(C2C(C)CC2)=O)CCC(F)(CNC(=O)Cn2ccc(=O)cc2)C1 C1(NC(CC2C(CC)C2(F)F)=O)CC12CCN(C(C1CC=CC(O)C1)=O)C2 C1(CC(=O)NCC#CCNC(c2[nH]cc(C#N)c2)=O)CC(O)C12CCC2 C1(CNC(C23OCC(CC)(C2)C3)=O)CN(C(=O)C=CCOC)CC(C)(C)C1 C1(C)(CCC(=O)NCC2(CNC(C(C)OCCC=C)=O)CCC2)CCC(=O)N1 CCCC(C(=O)N(C(c1ccccc1)CNC(C1CCCC(=O)C1)=O)C)OCC N1(C(CCCCCCC)=O)CCCC12CCC(NC(=O)C1=CCCS1)CC2 c1(C(N2CC(CNC(C(C)OC(C)=O)=O)C(C)C2)=O)ccc(S(N)(=O)=O)o1 N1(CCN(C)C(C2(N(C)C(C3COC(=O)N3)=O)CC2)=O)CCOCC1 C1(C(N2CC(N(C(=O)CN3CCCNC3=O)C)C(O)C2)=O)CCN(C)S1(=O)=O c1(C2(C(=O)NC(C(C)OCCOC)CO)CC2)ccc2c(c1)OCO2.C1C(=O)N1 N1(C(C(c2ccccc2F)C)=O)CC2(CC2)CC1CNC(C1CC2C=CC1O2)=O c1(C(=O)NC(C(C)NC(C2CC(F)C(=O)N2)=O)CO)cccc(O)c1Cl c1(C(c2ccco2)NC(Cn2cc(CCCC(=O)O)nn2)=O)cccc(Cl)c1 Cn1nc(C2CC2)nc1C(N1CCCC(C(N2CCC2C(C2CC2)C2CC2)=O)C1)=O c1(C(=O)NC)cn(C2CC2)nn1.C1(NC(C2(SC)CC2)=O)(CNC(N)=O)CCC1 c1(C(=O)NC(CC=C)CNC(c2c(C)[nH]c(C)c2C)=O)nccc2ccccc12 CCC(C(C)CN(C)C)NC(=O)C(C(C)C)NC(=O)CCc1nccn1C Cc1ccc2[nH]c(CN=C(NCC(C)(C)C)NCC(C)(C)C(F)(F)F)cc2c1 c1(NC(c2cnc(CC)s2)c2nnnn2C(C)(C)CC)cnc(C)c(C)c1 CCS(=O)(=O)CC(=O)NC(C)(C)C(C)NC(=O)CN(C)Cc1ccc(Cl)cc1 Cc1cc(OC(C)C(=O)NC2CC(C)N(C(c3occc3C)=O)C2)ccc1Cl N(C1CCCc2ccoc21)C(C(C)N(C(c1ccc(C)s1)=O)C)=O C1(NC(c2cc(C)ncn2)=O)CC2CC(NC(c3cn(C)cc3C)=O)C1C2 CC1CCC(C)(C(=O)NCc2csc(CNC(c3ccc(F)s3)=O)n2)C1 C(=O)(CCC(C)(F)F)N.C(=O)(CSC(F)F)N(C(C)C)CCO c1(C(=O)NC2(C3CN(C(c4conc4C4CC4)=O)C3)CC2)ccn2ncnc2c1 Cc1ccc(C(N2CC(=C(F)CNC(c3[nH]cnc3C)=O)C2)=O)c(N)c1 c1(CN2CC3N(C(C4=C(C)OCC4)=O)C(C3)C2)c(C)cc(C)cc1C c1(N(C)C)cccnc1C(N1CCOC(CNC(=O)Cc2ccc(Cl)cn2)C1)=O c1(CNC(C2CN(C(c3cnc(C)s3)=O)CC2C)=O)n[nH]c2ccccc12 CC1(C)CC(=O)CCC1C(N1CCCC(O)(CNC(=O)C=CCF)CC1)=O C1(CC(=O)Nc2n(C)c(CC(F)(F)F)nn2)CCCC2(CNC2)O1.c1cccs1 Cc1c(C=CC(=O)Nc2nnc(-c3ccc(Cl)cc3Cl)s2)cnn1C c1(C(=O)NCC2(COC)CN(C(=O)CC3(N4CCCC4)CC3)C2)cc(C)ccc1C Cc1cc(N)c(C(=O)NC2(CCCNC(c3ccon3)=O)CC2)cc1C N1(Cc2ccc(C)cc2OCc2ccccc2)Cc2ccccc2CC1C(C)C C#Cc1cnn(C(=O)NCC(CC(=O)N(C2CCOC2=O)C)OC)c1 C(=O)(C1CCCc2ncnn21)NC1CCN(S(c2c(C)c(F)ccc2)(=O)=O)CC1 C(=O)(C1Cc2ccc(C)cc21)N(CCN(C(CCOC(C)=O)=O)C)C N1(CCNC(CCC2(CNC(COCCCC)=O)CCC2)=O)CCC2CC12 Cc1ccc(C(N2C(CNC(C3(Cl)CC3(F)F)=O)CC3CC23)=O)cc1C N1(C(C2CCC(C)C2)=O)CCCC(C2CCCN(S(C)(=O)=O)C2)C1 Cc1ccc(F)c(CNc2cc(-c3cccc(C)n3)ccn2)c1 S(=O)(=O)(c1cccs1)NC1CCCN(C(c2c(F)cccc2F)C)C1 c1(CC)ccc(C(N2CCOC(CNC(c3cnccc3C)=O)C2)=O)cn1 CCCCC(=O)N(CC(C)NC(=O)CC1CC1C(F)(F)F)CC C1(CN(CCN(CC)CC)C(=O)Nc2ccccc2)CCCNC(=O)C1 C=CCC(C)(C)C(=O)NCC1CN(C(c2cc(C)n(C)n2)=O)C2CC12 C(=O)(C(C)(C)CCC(=O)N(CC(C)NC(=O)C=C(C)C(C)C)C)OC C(CCCCCN(C(=O)CC1CCC(C)(C)C1)C)NC(C(CC)F)=O Cc1ccc(C(C2(C)C(CN3CCN(CO)C(c4nc[nH]n4)C3)CC2)O)nc1O C1(CC=CCC(=O)NCC(C)NC(=O)CCNC(=O)C=CCl)CCCN1 c1(C(N2CC(F)(CNC(C(C)(C3CC3)OC)=O)C2)=O)cccc(C(C)C)n1 Cc1ncnc(C(=O)NCC(C)CNC(=O)COc2ccccc2Br)c1C c1(C(=O)NC2CN(C(C=C(COC)C)=O)CC(O)C2)cc(OC)cc2c1CCC2 c1(-n2cc(CSC)nn2)ccccc1C(=O)NC(C1CC12CCOC2)C1CCOC1 N1(C(CC2CCC(=O)C2)=O)CC2(CC2)CC1C(=O)NC(CO)CCCO c1(SC)cccc(NC(C2CCCN(C(=O)C(C)(C)O)C2)C)c1[N+](=O)[O-] c1(C(N2CCC(C(=O)NC(C(C(=O)OC)C)C)O2)=O)cc(C)ccc1F C(=O)(CC(C(F)F)NC(=O)C(C1CCCCC1)=O)NC(C(=O)OCC)C C1(NC(C2C=C(C)CS2)=O)CCCC(N(C(=O)CNc2ccccn2)C)C1 N1(C(C(CCC)Cl)=O)CCOCC12CCN(C(C1CCCOC1)=O)C2 c1(CCNC(=O)C(c2ccco2)NC(=O)CC2CCCN2C)c(CC)cnn1CC CCC(C)CCC(=O)N1CC(CNC(c2cccc(N(C)CC)n2)=O)(OC)C1 C(=O)(C(C)C(O)C(C)CC)NCC1CC(OC)CN1C(=O)C1=COCCC1 c1(CC)noc(C)c1C(=O)NC1CC(C)N(C(=O)COCC(=O)OC)C1 c1(N(C)C)c(F)cc(CN2CC(F)CC2C(N2CCS(=O)CC2)=O)cc1F c1(OC)ccc(O)cc1NC(c1cc(CCNC(=O)CCC2CC(C)C2)on1)=O C1(NC(CCN(C(=O)C=CCN(C)CC)CC=C)=O)COCCO1 c1(C(C(F)(F)F)CNC(=O)CN2CCC(c3cc[nH]n3)C2)ccc(Cl)cc1 C#Cc1cc(C(=O)NCCC2CCN(C(c3c[nH]c(=O)cn3)=O)C2)cc(Br)c1 C(=O)(C1=CCCCCC1)N1CCC(O)(C(C)NC(c2ccnn2CC2CC2)=O)C1 Cc1cc(OCC(=O)NCC#CCNC(c2ccsc2Cl)=O)no1 N1(C(C(=O)OCC)=O)CCC(Oc2cccc(Cl)c2)CC1.C12CC(C)N(C1)C2=O N1(C(C2N(C(COC(C)(C)C)=O)CC2)=O)CC2CC1CS2 c1(C(=O)OC)cccnc1Nc1ccsc1CO.c12c[nH]nc1C(=O)N2 C(C1COC(C)(C)O1)=CC(=O)NCCC(CNC(c1ccn(CC)c1C)=O)O C=C(C)C1OCCCC1C(=O)NC1COCC1NC(=O)COC1CCCCCC1 CCC(C)(C(=O)N(CCC(C(C)C)NC(=O)C(C)C)C)OC c1(C2(C(N3CC(O)(CNC(CC(C)SC)=O)C3)=O)CCC2)c(C)cccc1C C1(C(C)C)CN(C(=O)Cc2cc[nH]c2)CCN1C(=O)CN1CCCCCC1 c1(CNC(CCc2n(C(C(=O)OC)C)nnn2)(C)C2CC2)cnc(Br)c(F)c1 Cc1cc(C)c(S(=O)(=O)N2CCC23CC(c2ccccc2)C3)cc1[N+](=O)[O-] c1(CNC(c2n(C)cc(Nc3cn[nH]c3)c2)=O)ccc2cc(Br)ccc2c1 N1(C(=O)C2=CCCSC2)CCC2(CCCN(c3ncnc4cccc(F)c34)C2)C1 c1(C(=O)NC2CCN(C(C(CCOC)OC)=O)C2(C)C)c(C)ncn(C)c1=O C1(C(N2CCC(C)(CNC(CN(CCOC)C)=O)CC2)=O)CN2CCCC1CC2 C(=O)(C(CC(C)C)C(C)C)NC(CCC)CC(=O)N1CCC=C(F)C1 C(=O)(C(C)C(F)(F)C(F)F)NCC(CC=C)NC(c1cncn1C(C)C)=O c1(CCCCC)cn(CC(C2CN(C(c3nc(C(C)C)cs3)=O)C2)F)nn1 C1(NC(C=CC(C)(C)NC(c2ccn(CCF)n2)=O)=O)CN(C)CCN(C)C1 C1(C)(CSC)CN(C(=O)C=CC(C)NC(=O)CC2CSCCO2)C1 Cc1nc(C(=O)NC2(C)CN(C(C3CCCC(N(C)C)C3)=O)C2)c(C)s1 c1(C(N2CC(OCCNC(c3coc(Cl)n3)=O)C2)=O)cc2n(c1)CCC2 c1(C(=O)Nc2onc(C(=O)OCC)c2C)ccc(S(C)(=O)=O)o1 C=C(C)CC(C(=O)N1CCC12CN(C(=O)C=Cc1ccccc1F)C2)OC CCS(=O)(=O)C1CN(CCCOCC2CCCO2)C1.N12CCN(CC1)CCC2C CC(F)(F)C(C)(Cl)C(=O)NC(c1cccnc1)C(=O)O N1(C(C(C2CCC2)OC)=O)CCC2(CC1)CCN(C(=O)CC1CCC(O)CC1)C2 C1(C(N2CCCC(c3nc(C)c(C(C4CCC4)=O)o3)C2)=O)CC2CC2CC1C C1(C(N2C(C)(CC(C)C)CCC2)=O)CCOC2(CCN(CCF)CC2)C1 N1(C2CCN(CCC=CCC)C2)CC(C)OC2(CCCOC2)C1 c1(O)cnc(SC)nc1.C1(N(C(=O)CCOC2CC2)C)CC(C(=O)NC2CCC2)C1 CCCC(C(=O)N(CCCN(C)C(c1ccsc1)=O)C)c1ccccc1 C1(CCOC)(NC(C23C=CC(CC2)C3)=O)CCN(C(c2ccc(C(N)=O)o2)=O)C1 c1(CCC(N)=O)ccc(C(=O)NC2(CCNC(C3CCS(=O)(=O)N3)=O)CC2)cc1 CC1CCCC1(C)NC(c1ccn(CCNC(c2cnoc2C2CC2)=O)c1)=O C1(OC)CCN(C(=O)CCCNC(C2CCOC(=O)CC2)=O)C12CCC2 C(C)(C(C)C(=O)NCCOC1(C)CCC1)NC(c1nc(CC)oc1)=O CCCN=C(NCc1cccc(C(=O)OC)n1)N1CCSC(COC)C1 Cc1ccncc1C(c1nnnn1C1CC1)NC(C)CCN(C)C N1(C(C=CC(C)C)=O)CCCC1(C)C(N1CCCC(NC(N)=O)C1)=O C1(C(=O)OC)CN(C(=NCCCCl)NCc2nnc3n2CCC3)CC12CCC2 C(=O)(C1COc2ccccc21)N1CCCC(CCNc2nc(C)nc(O)c2C)C1 C1(c2n(CCCOC)nnn2)(Nc2ccccc2CN(C)C)CC2CCCCC12 N1(C(c2c(CC)nccc2)=O)CC(OC)CC1(C)CNC(=O)CN=S(C)(C)=O c1(C(=O)NCC2N(C(C(C(C)C)O)=O)C3CCC2C3)ccc2c(c1)NC(=O)CS2 c1(C(=O)NC2CCC(N(C(CCNC(=O)OCC)=O)C)C2)c(F)cc(C)cc1F C1(C(N(C2CCCN(C(c3c[nH]nc3C(C)C)=O)C2)CC)=O)CCCC(=O)N1 c1(C(=O)NCC2CN(C(=O)CC3CCS(=O)(=O)C3)CCO2)occ2c1CCCC2 c1(CNC(C2OCCN(Cc3cc(OC)ncc3Br)C2)=O)cc(F)cc(C#N)c1 c1(OC2CCN(C(COC)=O)C2)cc(N2CCOCC2)c(Cl)cc1Cl CC(C)(C)C#CC(=O)NCC1(C)CCN(C(C2COC(=O)O2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCCC2C1CCCN2C(=O)CCCC(N)=O n1(CCNC(CCCNC(=O)OC)=O)cnc(C)c1C.C1(C(=O)N)(CO)CC=CC1 C1(O)(CCC)CCN(C(C2CCC(CC)CC2)=O)CC1.c12coc(c1)CNC2=O c1(N(CCCN(C(CN(C(N)=O)C)=O)C2CCC=N2)CCN)ncnc2c1CCO2 c1(C(N(C)CC2CCN(C(=O)CO)CC2)=O)ccc(O)c(O)c1 Oc1ccc(N2CCCCC2)cc1NC1COCC1CC1CC1 C1(NC(CCCC(N)=O)=O)CC2(CCCN(C(C3CCN(CCF)C3)=O)C2)C1 N1(C(C2C(C)CCC2)=O)CCOC2(C1)CN(C(C1CC13CCC3)=O)C2 c1(C(=O)NCc2cn(CC(=O)NCc3cc(C)on3)nn2)ccc2cccnn12 c1(-n2c(-c3cc(C)sc3)nc(C3CC3)n2)cccc(S(C)(=O)=O)c1 C1(F)(CNC(C(C)C2CCCO2)=O)CCCN(C(=O)CCc2nncn2C)CC1 CN1C(=O)CCc2c(-c3nc(-c4ncccn4)nn3-c3cccnc3)cccc21 CN1CCN(CC(=O)N(CCC(C)(C)NC(=O)CC23COC(C)(C2)C3)C2CC2)CC1 C1(CNC(COCC(=O)OC)=O)CN(C(c2ccnn2CC(F)F)=O)CC12CC2 c1(NC(C2CC3CN(S(CC=C)(=O)=O)CC3C2)=O)cccc2c(O)nnc(O)c12 Cc1cc(F)cnc1C(N1CCC(C(=O)NCC2CCOC2C)C1(C)C)=O CC1C(NC(C2CSC2)=O)CCCN1C(C1CCCNS1(=O)=O)=O n1(CCCNC(c2cc(CNC(C3CC3C3CCCO3)=O)[nH]n2)=O)ncccc1=O N1(C(C(CC)(C)O)=O)CC(C(=O)Nc2cc(Br)cnc2F)C2(CC2)C1 C1(C(N2C(C(CC)C)CCC2)=O)COCCN(C(c2cc(C3CC3)no2)=O)C1 S(=O)(=O)(C1CCN(C(=O)NCc2nc(C(C)C)cs2)C1)NCC c1(NCC(C)NC(CCCOC)=O)ncnc2c1nnn2C(C)C C(C(=O)NCc1cccc(OC)c1)(C1=CCCSC1)N(CC(=C)C)C1CC1 c1(-n2cc(CC(CC)C(=O)NCC(c3ccccc3)=O)nn2)cc(C)nc(C)n1 C1(C(=O)Nc2ncc(OC)cc2F)CCCC12CCN(Cc1cc(C)n(C)n1)C2 c1(C(=O)NC2C(CNC(C(CC=C)C)=O)CC2)cn(C)c2ncccc12 C1(C(=O)NCC2(C)CCCN(c3ncnc(C)c3Br)C2)CCC(C2CCCO2)O1 Cc1c(C(N2CCC3(C2)CN(C(=O)CCCN=[N+]=[N-])C3)=O)ccc2n[nH]cc12 C1(CCC(=O)NCCC(C)N(C(=O)CCOCC(F)F)C)CCCOC1 C1(N(C)C)COCC1N=c1nccc(N(CCC#N)Cc2cccnc2)[nH]1 C1(n2cccn2)(CNC(=O)CC(F)F)CCN(C(=O)CC2CC2)CC1 C(N=c1nc(NCCCc2cn[nH]c2)c2cc(Cl)ccc2[nH]1)c1cn(C)[nH]c1=N Cc1cccc(OCCC(N2CCCC2CNC(C2CCSCC2)=O)=O)c1 N1(CC(=O)N(CCC(=O)N(C(C)CC(C)C)C)CC#C)CC2CCC1C2 N1(C(C(COC)NC(c2c(NC)cnnc2)=O)=O)CCCC(C)(C)C1C c1(C(=O)NCCC(C)N(C(CCSC)=O)C)ccc(COC(C)C)c(F)c1 c1(CC)cccc(OCC(=O)NC(C)CCNC(=O)C(C)(F)c2ccccc2)c1 c1(OC)ccc(CO)cc1.N12CCC(C1)N(CCC(=O)O)C(=O)NC2=O C=C(F)C1(CC(=O)NCC(CNC(c2ccnc(C)c2)=O)CO)CCC1 N1(CC)CC(NC(C2CC=CCN2C(c2cncc(C)c2)=O)=O)C(C)(C)C1 C1(O)(C(=O)NC(C)C(c2ccccc2)NC(c2csc(Cl)n2)=O)CC(F)(F)C1 CN1C(=O)NCC1C(=O)NC1CCCC1CNC(=O)CNC(N)=O Cc1ccc(N2CC(NC(=O)CC3CSCCN3)CC2=O)cc1C N1(CC(=O)NC2CN(C(c3cnoc3C3CC3)=O)C2)CCN2CCOCC2C1 C1(=CC(=O)N(C(CC(=O)N(C)CCc2ccc(O)cc2)=O)CC)CCCCC1(C)C C(C(=O)NCC1C=CCN1C(c1ccc(C#N)[nH]1)=O)(C(C)(C)C)N(C)C C(=O)(C(O)CC(F)(F)F)NC1CCC(NC(c2n[nH]c(C)c2Cl)=O)CC1 N1(C(C2(n3cc(C=CC)nn3)CC2)=O)CCC2(CC1)NC(=O)N(C)C2=O N1(C(C2C(C(C)C)C2)=O)CC2(C(=O)NC(C3CC4(CCC4)C3)C)CCC1CC2 c1(C(=O)NC(CCCC)CNC(=O)CNS(=O)(=O)NC)ccn2nncc2c1 N1(C(C(c2ccc(C)cc2)CC)=O)CCCC2(C1)CC(COC)(OC)C2 C1(NC(CS(CC)=O)=O)CC2CC1CN(C(=O)CSc1nc3ccccc3s1)C2 C(=O)(C(C)(CNC(C1CCC(=O)CC1)=O)CC)NCC(CC)(C)C C1(NC(C(CC=C)C)=O)CCC2CN(c3ncnc(=N)[nH]3)CCC2C1 CCC(C(=O)NCC1CC(F)CN1C(c1cc(C)n(C(C)C)c1)=O)C(C)C c1(C(C)C(N2CCC(C#N)C2)=O)cc(-c2ccc(F)cn2)cn2ccnc12 C1(N(CC(=O)NCCCCCNC(=O)CCn2ccnn2)C)CCCCC1F C(=O)(C1CCCc2ncnn21)NC1CN(C(CCC(C)c2ccccc2)=O)CC1C C1(NC(CCCOCCC)=O)CN(C(c2ccc(CC)c(F)c2)=O)CC2(CC2)C1 C1(CNC(c2cc(C)cc(C)c2)=O)CC2COCC2N1C(=O)CC1CCC(O)C1 Cc1cc(C(=O)N(C(CC(F)F)C(=O)NCc2cc(CO)on2)C)c(C)n1C CC1(C)CCC(C(=O)NC2CCC(NC(c3cc[nH]c3C3CC3)=O)CC2)O1 C1(NC(C(C)(C)OC)=O)CCCCC12CCN(C(=O)CSCCC(C)C)CC2 c1(-c2ccc(C(=O)NCCN(CCO)CCO)nc2)ccc2c(c1)C(=O)OC2 N1(C(C(C)OCC(C)C)=O)CCN(C(c2ccn(C(F)(F)F)n2)=O)CC1 C(=O)(CC(C)CC(C)C)NCC1N(C(c2c(CC)ccs2)=O)CC(F)(F)C1 C1(NC(Cc2ccc(C)o2)=O)CCN(C(=O)CCn2cc(Cl)cn2)CC1C c1(CCCCOC(C)(C)C)nc(-c2nc[nH]n2)nn1C1CCC1 CC1(C)OCCC1C(=O)NCc1ncc(C(=O)NOCc2nc[nH]n2)cn1 N1(CCC)CC2(CCC2)C1C1CCN(C(C2(C(=O)OCC)CC2)=O)CC1 C1(C(N2CCC(N(C(c3cn(CCOC)nn3)=O)C)C2)=O)OCC2COCCC12 C1(NC(COC)=O)CCN(C(C2CCSC2)=O)CCC1(F)F Cc1cc(Br)cc(F)c1NC(c1coc(Br)n1)=O Cc1[nH]nc2cc(C(=O)NCC(C)(C(C)C)NC(c3cnc(S)[nH]3)=O)ccc12 C1(NC(c2c(C)cc(OC)cc2F)=O)CN(C(=O)C(C)=C(C)C)C2(CCOC2)C1 CC(C)CC(C(=O)NCCC1CCCN(C(c2cc(C#N)cs2)=O)CC1)C(C)C Cc1cc2ccccc2nc1C(N1CCCC2(C1)CN(C(C1CC1C)=O)C2)=O C12(C(N3CCC(CC)(NC(C4CCC(CC)CC4)=O)C3)=O)CCC(F)(CC1)CC2 c1(CN(C)CC2CCN(C(C(COC)C)=O)CC2)ccc(C(=O)O)cc1F C1(C(=O)NCC(CC)NC(c2scc3c2OCCO3)=O)CCCCCS1(=O)=O Cn1nc(CNC(c2csnn2)=O)cc1C(=O)NC1CC(O)C1(C)C c1(-n2c(CCSc3cccs3)nc(C(CC)O)n2)cc(C)nc(C)c1 N1(CC(N2CCC(CC(=O)NC3(C4CCC4)CC3)C2)=O)CCOCC1=O CC1(CNC(c2cscn2)=O)CCN(C(c2cc(C(N)=O)co2)=O)CC1 N1(C(C2(C(=O)OCC)CC2C)=O)CCC(CCNC(=O)CCCSC)C1 c1(C(N(CCCN(C(=O)C(F)(F)C2CC2)C)C)=O)cc(S(N)(=O)=O)ccc1O c1(CC)ccc(C(C)C(=O)N(CCCNC(=O)Cc2csc(C)c2)CC)cc1 c1(C(N2CC=CC(NC(CC(CC)C(C)C)=O)C2)=O)cc(=O)c2ccccc2o1 C1(C)(C(=O)NC(CN(C(=O)CN2CSCC2=O)CC)C)COc2ccccc2O1 N1(C(CN(C(CN(CC)CC2CC2)=O)C2CC2)=O)CCCC(CCO)C1 N1(C(C23CN(C(CCC(C)C)=O)C(C2)CO3)=O)CCC(C2(C)CC2)CC1 N1(C(c2cccc(Br)c2N)C(=O)Nc2nnn(C)n2)CCC(O)C(F)(F)C1 c1(C(N2CCC(C)(CNC(C3CCCN3C=O)=O)C2)=O)noc2ccccc12 N1(C(C(C)=C2CCC2)=O)CCCC(C(C)NC(=O)COc2ccc(F)nc2)C1 Cc1cc(C(N2CC3CC2C3NC(=O)C(O)C2CC2)=O)cc2nn[nH]c12 c1(OC)ccccc1C(C)CC(=O)NCCCCCN(C)C(c1sccc1F)=O N1(C(c2c(C(C)C)c[nH]c2)=O)CCCC(NC(C2CC3CCC2O3)=O)C1 C1(CNC(C(C)OCCC#C)=O)CCCCC1NC(c1ccnnc1C)=O C(=O)(C(F)(F)CO)NC1(CNC(=O)CCc2nc(C3CCOCC3)no2)CC1 N1(C(CN(C)Cc2ccc(OCC)cc2)=O)CCN(C(C2CC23CC3)=O)CC1C CC(C)C(C)(CNC(=O)C=CC(C)NC(c1csnc1Cl)=O)C(C)C c1(C(=O)NCC2(O)CCCN(C(CC)=O)C2)cc2c(o1)CCCNC2 CC1(c2cn(C3(C(=O)OC4CCCO4)CC3)nn2)CCN(C(N)=O)C1 CCC(CC(=O)N(C)CC1CCCC1NC(=O)CN1CCCNC1=O)CC(C)C CCC(CC(F)(F)F)C(=O)NC1CN(C(C2(CN(C)C)CCCC2)=O)CC1OC c1(N(C(C)COC)CC=C)ccnc2ccsc12 Cn1cc(C(F)=CC(=O)NCCNC(C2CC2C(F)(F)F)=O)cn1 S(=O)(=O)(c1cccnc1N1CCC2CCC(C1)N2C)N(CCCC(C)C)C S1(=O)(=O)CCC(=O)N2CCC2CNC(=O)CO1.c1(OCC)ccc(C)cc1 c1(C(=O)NCC=CCNC(C2C(OC)CC2)=O)sc(-c2ncccn2)nc1C c1(C(C)NC(c2c(NC(C=CC(CC)C)=O)ccs2)=O)ccccc1C C1(NC(C23CC(CN(C(C(C(C)C)C4CCC4)=O)C2)C3)=O)CC2CC1CC2(C)O c1(CNC(CC(=O)NCC2(NC3CC3)CC2)=O)cccc(N2CCCC2)c1 c1(CCC)c(C(=O)NCCNC(=O)CCC2CC2C)cnn1-c1cccc(Cl)c1 N1(C(c2cc(OC)no2)=O)CCC2CN(C(=O)CCc3ncc[nH]3)C2C1 c1(CCC(C)=O)cn(C2CCC(CC(N3CCOCC3)=O)C2)nn1 O=C(C1=NN(c2ccccn2)C(=O)C1)N(C1CC1)CC1CCCOC1 c1(OC)ccc(C(=O)NC2CC2CNC(=O)CCc2cn(C)cn2)cn1 C(=O)(C1CCCc2nncn21)NC1CC2N(C(CCCN=[N+]=[N-])=O)C(CC2)C1 c1(OC)ccc(CC(=O)N(CC(C)NC(C2(CO)CCC2)=O)C)cc1F c1(C(C(N2C(C(C)NC(c3ncoc3C(F)F)=O)CCC2)=O)O)ccc(Cl)cc1 c1(C(N2C3CC(N(C(C(C)=O)=O)C)CC2CC3)=O)ccc2c(c1)nnn2C C(=O)(CCCS(=O)(=O)N1CCOCC1)Nc1sc(C)c(C2CCOC2)n1 Cc1nsc(C(=O)NC(C)CC(C)NC(=O)C=CC2CCC2)c1N c1(NC(=O)NCc2c(CC)ocn2)cccc(S(=O)(=O)N(C)OC)c1 NS(=O)(=O)CCN(CCC(=O)NCC1CCCCO1)C(C1CCCC1)C n1(CC(=O)NCC(C)NC(c2ccccc2CN(C)C)=O)ncn(C)c1=O N1(C(C2N(C(CNC(C)=O)=O)CSC2)=O)CC(=O)NCC1C(N)=O c1(C(=O)NCC(CC)NC(=O)Cc2ccc(Cl)nc2)cc(C)nn1C c1(C(=O)NC2CC(OC)CN(C(C3CCO3)=O)C2)cc(F)cc2ccoc12 C=CCC(C)(CO)CN=c1[nH]c(=N)[nH]c(=NCc2nnc(O)o2)[nH]1 c1(C(N2CC(O)(CCNC(COCC)=O)C2)=O)ccc(Cl)c2ccccc12 c1(OC)ccc(Br)cc1C(c1nnnn1C(C)C)NC1C=CCCC1 n1(CC(=O)NC2C(C)N(C(=O)CC3CCC(F)(F)CO3)CC2)ncc(O)nc1=O c1(N(C)CC2CCCN(C)C2)nc(=NCC2(CO)CCCO2)[nH]c2ncn(C)c12 CCCC(N=c1[nH]c(=NC(C)c2cncs2)[nH]c2c1CSC2)C1CCCC1 Cc1ccc(NC23CNCC2C3)cc1OCC(F)F Cc1cccc2c(C(=O)NCCCC(C)NC(=O)COc3ccccc3)n[nH]c12 C1(C(=O)NCCC2(O)CN(C(CCC(C)OC)=O)C2)CC2(CC(C)=NO2)C1 c1(C(=O)NCC2C(NC(CCNC(COCC)=O)=O)C2)cc2sc(C)cc2s1 c1(C(=O)NC(CCNC(c2nc(C)nc(O)c2)=O)C)ccc(Cl)c(C)c1Cl C1(OC)CCC2CN(Cc3cn(-c4cc(Br)c(F)cc4F)nn3)CC12 c1(CC(=O)NC2CC(C(=O)NCC3(CO)CCC3)C2)c(O)ncnc1O c1(CC(=O)NCC=C2CCN(C(COC)=O)CC2)ccc(Cl)c(Cl)c1C Cc1cn2c(n1)CC(C(=O)N(CCC(C)(C)NC(C1CCOC1C1CC1)=O)C)C2 C1(OC)CC(NC(c2ccc3c(c2)OCO3)=O)C12CCNCC2 Cc1cc(C(=O)NCC2(NC(=O)C(CO)C(C)C)CCOCC2)c(N)c(Cl)c1 C1(CC)CCCN(C(c2ncccc2COC)=O)C1C(N(C)CCO)=O C1(NC(C(C)N(C(=O)CC2CCOC2(C)C)C)=O)CCCCCC1C c1(C(N2C(C(=O)NCC3CCC(O)C3)CC3(CC3)C2)=O)cc(I)ccc1[N+](=O)[O-] N1(c2cccc(N3CCN(C(c4sc(C)c(O)n4)=O)CC3)c2)CC(C)OC(C)C1 c1(OCC)cnc(OC)c(C(F)F)c1.c12noc(n1)CNC2C C1(C(=O)NCC2C(C)CCN(C(=O)C(=O)NCC3CC3)C2)CCC12CCOCC2 c1(C(N2C(C)CC(NC(c3ccc(CC)cn3)=O)C2)=O)ccc2nc(O)sc2c1 c1(C(N2CC(N(c3ncccn3)C)C2)=O)cc2cc(F)c(F)cc2[nH]1 C1(CNC(CC(C)(F)F)=O)CCCN(C(C2(CO)CC2(F)F)=O)CC1 c1(C(=O)NCCCNC(CCNC(COC)=O)=O)ccc(-n2cccc2)nc1 Cc1ccc(NC(=O)C(C)Nc2cc(-c3ccc(F)cc3)n[nH]2)c(C)c1 N1(C(C2(C)CCC(C)C2)=O)CCC(C)N(C(C23CC(C)(C2)OC32CCC2)=O)CC1 C(c1ccccc1Cl)=C(C(=O)NC(CCOC)CNC(C1CC=CCC1C)=O)C C1(CNC(=O)COCc2nc[nH]n2)CN(C2CC2)CC1(F)CO.c1cnc(CO)s1 C1(C(=O)NCC(CC)OC)CC(C)CCN1C(=O)CCCOC(C)(C)C N1(C(c2cc(C#N)sc2)=O)CC(NC(c2cccc3cc[nH]c23)=O)C(C2CC2)C1 C1(CC)(NC(c2oc(C)cc2C)=O)CCN(c2nc(C3CCCCC3)ns2)CC1 C=Cn1nncc1C(N1CCC(CCN(C(=O)CC2CC3(CC3)CO2)C)CC1)=O CCCC(CC)C(=O)N1CCC(CCNC(=O)CCCC#N)C1 c1(C(=O)NC(CCNC(CCn2ncc(C)c2)=O)C(C)C)cc(C)c(CO)cn1 C=CCC(CC)C(=O)N1CCN(C(c2ccc(C3CCC3)nc2)=O)C(C)C1 C1(C(=O)OCC)CC2CCC1N(Cc1ccccc1)C2.C12CCCC1ON2 Cc1ccncc1C=CC(=O)NC1CC2(C1)CC2F.C1C=CCO1 C1(NC(c2ccnnc2)=O)CC(CO)N(C(C2CCCOC2)=O)C1 CCC(C)C(C)C(=O)NC(C1CCCN(Cc2cnc(C)o2)C1)C C1(CN(C(CSCCOC)=O)C)CCN(C(c2cc(-c3ccccc3)[nH]n2)=O)C1 C1(C(=O)NC2(C(O)CO)CC2)C=CC(C(=O)NCCC2CCSC2)C1 C12(C(=O)NCC(CC(C)C)NC(CC(CC)C)=O)CCC(N(C)C)(CC1)CC2 c1(C(N2CC(C)(NC(C3CCC(C(F)(F)F)C3)=O)C2)=O)cn2ccnc2s1 Cc1ncn(C)c1C(=O)NC1CN(C(C2COCCN2C)=O)CC1C N1(C(CC(C(C)C)C)=O)CC2CCC1C(NC(=O)CN(C1CCCCCC1)C)C2 C1(c2scc(C)n2)COCCN1C(=O)NCc1cccc(Cl)n1 c1(NC(c2cnsc2)C)nc2ccccc2nc1N1CCC(OCC2CCCO2)C1 CCCC(C)(CC)C(=O)NCC1(OC)CCN(C(c2cc(C)cnc2N)=O)CC1 c1(C(N(C)CC2CCCN2C(=O)CC2CCC(=O)CC2)=O)c(F)ccc(N)c1F CS(=O)(=NC(=O)c1nc2ccccc2s1)c1ccc(Cl)c(Cl)c1 Cc1ncc(CN(C(c2ccc(Cl)o2)C(=O)NCC(C)C)C)n1C N1(N(C(C)(C)C)C)CCCC(OCc2cn(CCCCF)nn2)C1.C=O c1(C(C)=O)cc(C(=O)NCCCN2CCN(C(C3CC(O)C3)=O)CC2)ccc1C N1(C(c2c(C)n[nH]c2)=O)C2CCC(C1C(N1CCC(C)C(O)C1)=O)C(F)(F)C2 C(=O)(CC(C)C(=O)NC1CCCCC1CC(=O)NCCC1CCCCC1O)OC c1(C(N2CC(NC(=O)COC3CC(CF)C3)C(O)C2)=O)ccc(Cl)c(Cl)c1 C#CC1(C(=O)NCC2CC=CCC2)CN(C(C2CC(OC3CC3)C2)=O)C1 c1(C(=O)NC2(COC)CN(C(=O)C=CC(=O)N(C)C)C2)ccc(Cl)cn1 C1(C)(C(=O)NCC2(C(C)NC(C3CCCCC3O)=O)CC2)CCC(C)C1(C)C c1(C(=O)NC2C(C)CCN(C(C3(CO)CCC3)=O)C2)ccc2c(c1)C(=O)C(=O)N2 C1(C(=O)NC2CCCC(NC(C(C)=C(CC)C)=O)C2)Cc2ccc(OC)nc2N1 C1(c2ccccc2)CCN(CCCSCCN2CC3CCCC2C3)C12CC2 C(C(=O)NCC1(NC(=O)Cc2ccc(O)c(Cl)c2)CCOC1)(C(C)(C)C)N(C)C c1(CN2CC(C)(C(=O)O)C(C(F)(F)F)C2)ccc2cc(Br)ccc2n1 Cc1nc(O)c(C(=O)NC(C2CN(C(C3(CCF)CC3)=O)C2)C)cc1C(F)(F)F N1(C(C(c2ccccc2)NC(=O)C=CC=C)=O)CCCCCC(=CC=CCC)C1 c1(NC(CCN(CCC)C(=O)C2CC2)=O)ccccc1S(=O)(=O)NC(C)CC C1(C(=O)NCC2N(C(C)=O)CCC2)CN(C(=O)CNC=O)CCN1C C(C(O)C(=O)NC(C)CC1CN(C(c2cc(-c3ccccc3)ns2)=O)C1)=CC C1(CC)CN(C)CCN1C(C1CC(OC)CCN1C(C1C2(CC2)C12CC2)=O)=O c1(NS(C)(=O)=O)ccc(C(=O)NCC2CCN2C(c2ccc(Cl)cn2)=O)cc1 C12(NC(CN(C)CC)=O)CC1CN(C(c1cc(C(=O)OC(C)C)on1)=O)C2 N1(C(C2(C)CCCC2O)=O)CCC2(CC1)CNCc1ccccc1O2 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(C(N2CCOCC2(C)C)=O)CC(OC)C1 CC1(C)CCC(C(=O)NCC2CCCC3CC23)(NC(=O)Cc2cncc(F)c2)C1 C(=O)(CC(C)(C)c1cccs1)NCC1N(C(C(CC)c2ccco2)=O)CC=C1 c1(C(=O)NC2CC(CNC(C3(CC#C)CCCO3)=O)C2)cncc(C)n1 c1(C(N2C(C)CN(C(CCCOCC)=O)C(C)C2)=O)ccc(S(=O)C2CC2)cc1 Cc1cc2[nH]c(=O)c(C(N3CCC(N(C)C(c4cnc(S)n4C)=O)C3)=O)cn2n1 c1(C(=O)NC2C(NC(c3c(C)sc(O)n3)=O)CC2)cnc2c(F)c(F)ccc2c1 C1(C(N(CCC#C)CCO)=O)CN(C(c2sccc2C#N)=O)CC1(C)C C1(NC(C(c2cccc(OC)c2)C)=O)CCN(C(=O)C=CCF)C1(C)C C(=O)(C(CC)C(C)(C)CC)NCCc1c(C(=O)NCCOCCCCC)c[nH]n1 C1(C(N(C)CC2OCCN(C(CN(C(C)C)C)=O)C2)=O)CCc2c[nH]nc2C1 C(C(CC(F)(F)F)NC(=O)C(c1cccc(O)c1)C)NC(c1c(C)sc(O)n1)=O c1(C(=O)NCCC2N(C(C(C)O)=O)CCSC2)c(Cl)c2ccc(Cl)cc2n1C c1(C(N2CCCC(C)(C(=O)NCCSC)C2)=O)ccc(C#N)c(C)c1 c1(C(=O)NC2CC(C)(OC)C2)cc(C(N2CCCC2C(=O)NC)=O)ccc1Cl CCC(CC(=O)N1CCN(c2nccc(NC(C)C(=O)OC)n2)CC1)C1CCC1 Cc1ccc(C#N)cc1C(=O)NCC(CC(F)(F)F)NC(c1ccnn1C(F)F)=O c1(C(=O)NCCN(C(C2CCC(CCO)CC2)=O)CC)cnccc1OC C1(C(N2CC(O)(CN(C)C(C3CCC3)=O)C2)=O)C2CCOCC12 S(=O)(=O)(c1ccc2c(c1)CCO2)N1CCC(N(C(C(CC(C)C)O)=O)C)C1 CC1COCCN1CC(=O)O.C(=O)CCCn1cc(CC(C)(C)C)nn1 CC1CCC=C1C(=O)NCCN(C)CCOCc1cccc(F)c1O C1(C(=O)NCCOCCCNC(c2cnn[nH]2)=O)COc2cc(Cl)ccc2C1 c1(C(=O)Nc2nc(Br)cs2)cc2n(n1)CCN(Cc1cc(Cl)ncc1Br)C2 c1(C(N(CC(=O)O)Cc2cn(CCCCC=C)nn2)=O)cc2cccn2cn1 c1(C(=O)NC2(C)CCN(C(=O)CCc3cncs3)C2)ccc(N)c(Cl)c1O CN(CC1(S(C)(=O)=O)CCC1)N1CCOCC1C1CCC1.C(C)(C)(C)N(CCO)CCO N(C(=NCCF)N1CCC2=C(CCCC2)C1)Cc1cn2cccc(C)c2n1 c1(C(N2CCCCC(CNC(=O)CCCCCF)C2)=O)cnc2n1CCS2 C1(CCNC(CCc2nc(C)sc2)=O)CN(C(c2ccc(F)o2)=O)CC1C N1(C(C(Cc2ccoc2)NC(C(CC=CC)C)=O)=O)CC(O)C(O)C1CO Cc1cccc(F)c1C(N1CCC2(CC2C(N2CC(n3cccn3)C2)=O)C1)=O c1(C(=O)NCC(C)(CO)NC(c2ccc(F)cc2)=O)ccc(C#CC2CC2)cc1 C12CCC(C1)NC(=O)C2.N1(C(C2(CCC)CC2)=O)CC(O)(c2nn[nH]n2)C1 N1(C(C(C)Cn2cccn2)=O)CC2CC(C1)N2C(=O)CCC(C)(F)F Cc1ccc(C(=O)NCC2CC2CNC(c2cc(=O)cc[nH]2)=O)c(F)c1Cl CC1(C(=O)NCC2CN(C(=O)CN3CCC(F)(F)C3)C2)CCCC1O c1(C(=O)NC2(C)C(CC)CCC2)ccc(OCC(C)C)c(Br)c1 C(=O)(C(O)Cn1cncn1)NC(C1CCCC1)C.C1(=O)CCOCCN1 CC(C)CCC(F)C(=O)N1CC2(C1)CN(C(c1ccc(F)c(O)c1F)=O)C2 N1(C(CC2(COC)CC2)=O)CCC2(CC(NC(c3cn(C)nc3C)=O)CO2)C1 N1(C(CCOCC#C)=O)CCN(C(=O)C(C)NC(N)=O)CC1CCCC CC1(NC(=O)C2=CCSC2)CCN(C(C2(Cc3cccs3)CCCC2)=O)CC1 C1(NC(c2cccn(O)c2=O)=O)CC2CN(C(c3ccon3)=O)CC12 C1(NC(Cn2nnc(C)n2)=O)CCN(CCC2CCCC2(F)F)CC1C N1(C(CCC(C)OCC)=O)CC2(C1)CN(C(C1(F)CC=CCC1)=O)C2 C1(NC(c2ncoc2C2CC2)=O)CC2(CCCN(C(C3(C(F)F)CCC3)=O)C2)C1 C(C1=NOC(C)C1)NC(c1nc(CNC(C2C(CC)C2)=O)oc1)=O Cc1cc(C(N2CCC(NC(c3occc3Cl)=O)C2)=O)c(F)c(Br)c1 c1(C(=O)NC2CC(NC(=O)CCn3cnnn3)CC2O)csc2ccccc12 C1(C(N(C(CCC(C)C)C)C)=O)CC12CCN(C(C1CC(N(C)C)C1)=O)CC2 CCCCCCC(C)n1nc(CC(C)C)nc1-c1cnsn1 Cc1cc2ccc(C(N3CCOCC3CNC(=O)CC(C)CN(C)C)=O)cn2c1 C(C(C)C)(C(O)C(=O)N1CCOC(C(=O)NC(c2nccs2)C)C1)OC c1(C(=O)NC2CC(C(C(=O)NC(C=CC)C)F)C2)ccn(C(C)C)n1 N1(C(CCNC(c2ccsc2)=O)=O)CCOC(CNC(c2cncnc2)=O)C1 c1(OC)cc(C)c(C(=O)NC(C)(C)CCNC(C23CC2COC3(C)C)=O)cn1 c1(CCC)nc(C)c(C(=O)NC2CN(C(=O)CC(C)F)CC2C(F)(F)F)s1 N1(C(C=CC(C)NC(C(C(C)C)NC(C)=O)=O)=O)CCC2(COC(C)C2)C1 CC(C)CC(CNC(C1CCC(N(C)C)C1)=O)C(=O)NC1CC2CCCCCC12 C1(C(=O)OC)(NC(=O)C(CCCC(=O)Nc2ncn(C)n2)N(C)C)CCCCC1 C(N=c1[nH]c2c(c(=NCc3nc4ccccc4o3)[nH]1)COC2)CCCS(N)(=O)=O c1(C(=O)NCC2CCN(C(C(C)OCCC#C)=O)C2)ccc(C)c(Br)c1N c1(C(N2CC(CNC(CC(COC)(C)C)=O)C(C)C2)=O)cc2c[nH]cnc-2n1 C1(O)(CCNC(C(C)n2ccnn2)=O)CCCN(C(c2cc(Cl)c[nH]2)=O)C1 C(=O)(C1=C2CCCN=C2NN1)N(CCNC(C1CCC1(C)C)=O)CC c1(NC(CN2CC3C(c4nc(C)[nH]n4)(C3)C2)=O)ccc(Cl)c(F)c1 C(=O)(C1Cc2ccccc21)NC12CN(C(c3c(C)cccc3Cl)=O)C(C1)C2 c1(N2CCC(CNC(CC(C(=C)C)OCC)=O)(CO)C2)ncccc1S(C)(=O)=O N1(C(C2(NC(C3C(C)OCCC3)=O)CCOCC2)=O)CCN2CCC1C2 c1(CC)cc(N2CCC(NC(c3ccc(C(F)F)nc3)=O)C(O)C2)nc(C)n1 C1(NC(c2c(O)cncc2F)=O)CC(O)CN(C(C2CCC2)=O)C1 C12(C(N3CC(O)(CNC(c4occ(C(N)=O)c4)=O)C3)=O)CCC(CO)(CC1)C2 O=S1(=O)CCC2(CCN(S(=O)(=O)c3cc(F)c(F)c(F)c3)CCO2)C1 C1(CNC(C(N2CCCCCC2)C)=O)CC2CCC1N2C(C1(F)CCC1)=O S(=O)(=O)(c1ccc(NC2CCCC(C)C2C)cc1)N(C)Cc1cc(C)cs1 N1(C(C2CC(CCNC(CCCN(C)C)=O)C2)=O)CCC(O)C1(C)C C1(c2nnnn2CCC2CC2)(SCC)CC2CCN(C2)C1.c12cccc(c1)CN2 C(CCCCCNC(C1CCC(C(N)=O)C1)=O)NC(c1cc(C)no1)=O N1(C(COc2ccc(C)s2)=O)CCN(C(c2cccc(-n3cccc3)c2)=O)CC1 N1(C(c2c(C)nc(C)s2)=O)CC2CCC(C(N3CC(F)C(F)C3)=O)(C2)C1 S(=O)(=O)(c1ccccc1)NCCC(=O)NCC(CNC(C(C)CO)=O)(C)O CCC(C)CC(=O)C(=O)N1CC2CC2C1C(=O)NC(C)C(C)(C)C N1(C2CCN(C(c3ccc(SC)o3)=O)C2)CCN(C(=O)CC(C)(C)C)CC1 CCC(CCC(=O)Nc1ccc[n+]([O-])c1)NC(C1CCOC1=O)=O N1(C(c2n(CC)ccc2)=O)CCCCC1CN(C(=O)C(C)(C)c1ccns1)C c1(NC(C23C(CN(C(C(CC)CC)=O)C2)C3)=O)cc(O)ccc1C c1(C(=O)NC2CCN(C(=O)CC3CCC4CC4C3)C2)ccn(CCO)c(=O)c1 Cc1cc(C)c(C(=O)NC(C2CN(C(=O)CCCNC(N)=O)CCO2)C)c(C)c1 C1(C)(NC(C2CC(O)(CC#C)C2)=O)CCCN(C(c2ccccc2OC)=O)C1 O=C(CC1=NNC(=O)C1)N(C1CCCC1)CCNC(c1ccc2cnsc2c1)=O N1(C(C(C(C)C)O)=O)CCN(C(C2(n3cnnn3)CC2)=O)C(C)C1 C(=O)(CC(C)C(=O)OC)N(CCC(N1CCCC1(C)COC)=O)CC#C c1(C(=O)NCC2CC(O)(CNC(C3CCO3)=O)C2)cc(F)cc2ccccc12 CCCCCC(=O)N1CCC(=CCNC(c2cc(Br)co2)=O)CC1 c1(N2CCC(O)(CC(C)NC(C3CCCC3C)=O)C2)ccnc(C2CC2)n1 c1(NC(CNC(CNC(CCSCC)=O)=O)CSC)c(F)cccc1F C1(C(=O)NCC(CC(C)C)(C)NC(C23CC(C)(C2)C3)=O)CNC(=O)CC1(C)C c1(CNC(=O)NC(c2nccs2)CC)ccc(OCC(N)=O)cc1 c1(C(N2CC(NC(C3CCCC(C)(C)C3)=O)C2)=O)cc([N+](=O)[O-])c(F)cc1Cl N1(C(CC(=C)C)=O)CCC2CN(C(c3cc(C)c(C(N)=O)cn3)=O)CC12 c1(C(=O)NCC(C)(C2CC2)NC(=O)C#CC2CC2)ccn2nccc2n1 N1(CCNC(=O)NCCC(CNC(=O)OC(C)(C)C)(C)C)CCc2sccc2C1 c1(C(N(CCCNC(C(N2CC(C)C2)C)=O)CCO)=O)c[nH]cc1Br c1(CN2CC(CC(=O)Nc3c[nH]nc3Br)C2)cnc(Cl)c(F)c1 N1(C(C2C(C)(C)C2(C)C)=O)CCN2C(=O)C(NC(c3cc(C#N)c[nH]3)=O)CC2C1 C(=O)(C1=COc2ccccc2O1)N(C(CNC(C1CCOC1)=O)C1CC1)C C1(C(N2CCC(NC(c3c(C)nc(C)[nH]3)=O)C(F)C2)=O)CC2C=CC1C21CC1 c1(OC)cncc(C=CC(N2CC3CC2C3CNC(=O)CC2CCC2)=O)c1 C1(C)(COC)CN(C(=O)CN(C(=O)Cc2cnc(C)s2)C(C)C)C1 c1(OC)cc(NC(=O)NC2CCC3CCC2C3)c(OC)c(C)c1OC C(=O)(C1=CC(C)(C)C1)OC(C)CCC(=O)NC(C12CC(CO1)C2(C)C)=O N1(C(C(C)S)=O)CCN(c2ccc(S(=O)(=O)N3CC4CC4C3)cn2)CC12CC2 c1(CC)noc(C(N2CCCCC2CNC(=O)COCc2nccn2C)=O)c1C Cn1cnc2c(C(=O)NCC(CC3CCOC3)C(=O)O)cccc12 C1(C(=O)NC2CCCN(C(CC3N(C)CCCC3)=O)C2)CN2CCC1CC2 Cc1onc(Br)c1C(=O)NC1CCOCC1NC(c1ncc(F)cn1)=O c1(C(=O)OC)cc(CN2CCN(C(c3ccccc3)=O)C3(CC3)C2)c(C)c(C)c1 C1(C(=O)NCC(C)(C)CO)(CC)CCCN(C(c2cncc(NC)c2)=O)C1 c1(CN(CCC(F)(F)F)C2CC2)ccnc(NCC(=O)NC)c1 c1(C(=O)NC(c2cn(CC(O)CO)nn2)CCC)cnc2[nH]c(O)nc2c1 N1(CC)C(=O)CCC1C(N1CC(=CC(=O)NCCNC(=O)C2CC2)C(C(F)(F)F)C1)=O c1(C(N(CCC)CCNC(C2CCCC2(F)F)=O)=O)c[nH]c2c(C)cccc12 c1(C(COC)NC(CC(C)(C)n2cccn2)=O)cn(C(C)(C)C)nn1 C1(C(=O)NC(C(=O)NC2CC(O)C2)C2CCCC2)CC2(CCCO2)C1 N1(C(c2ccnc(OC)c2Br)=O)CCC2(O)CCCCC12 C1(OC)(CNC(C2(C3CC3)CC2)=O)CCN(C(c2cc(C3CC3)no2)=O)CC1 C(=O)(CC(C)(C)CSC)NC1C(NS(CCC)(=O)=O)CCCC1 c1(C(=O)NCC=CCNC(C(CCC)(C)C)=O)cc2c(Br)ccc(F)c2[nH]1 C=CC1(C(N2CCN(C)CC2C(C)C)=O)CCN(C(=O)C(=O)NCC)C1 c1(CC)ccsc1C(N1CCCC1CN(C(c1cc(C2CC2)cs1)=O)CC)=O N1(C(c2nccc(CC)c2)=O)CCC(CO)(NC(c2ccc(C)nc2Cl)=O)CC1 CC1CN(c2ncc(F)c(-c3cccs3)n2)CCCN1CC(F)(F)F C1(C(=O)NCC(CC)NC(C2CCN(C)C(=O)C2)=O)Cc2ccc(C)cc2S1 C1(NC(CC)=O)COC2(CCN(C(=O)Cc3csc(N4CCCCC4)n3)C2)C1 C(=O)(C1CCCc2ccccc21)N1CC(F)(CNC(c2c(OC)ccs2)=O)C1 c1(C(=O)NC2(C)CC(NC(C(C3CCC3)OC)=O)C2)cc(C(N)=O)cn1C c1(N(C(c2c(CC)con2)C(=O)NCCOCC2CC2)C)ccc2cnccc2c1 N1(C(CNC(c2ccc(C)s2)=O)=O)CC2CCC1C(NC(c1oc(C)cc1C)=O)C2 c1(C(N2CC(OC)CC(C(N)=O)C2)C(=O)NC)nn(C)c2c1CCC2 C(=O)(C1CCc2nccn21)NC(C1(C(=O)NC(C(C)C)c2ncc[nH]2)CC1)C C(=O)(C1CCc2ccccc21)NC1CCCC(NC(c2cn(C)nc2Cl)=O)C1 CC1CN(C(c2cnc(O)s2)=O)CCN(C(C2(C)CCCOC2)=O)C1 C(CCC(=O)N1CC(CNC(c2conc2C(F)F)=O)C1)NC(N)=O C1(CN2CC(C#N)OCC2)CC2(CCOCC2)CO1 c1(C2(C(=O)NCC(CNC(C3C(OCC)C3)=O)(C)C)CCCC2)ccc(C)cc1 Cc1snnc1C(N1CCC(C2CCCN2C(=O)CN(C)C)C1)=O C1(NC(C=Cc2c(C)ccs2)=O)CN(C(=O)C(C)N2CCC2)CCC1F Cc1cc(-c2ccnc(N3CCSCC3CO)c2)c(F)cc1F C=CCC(CNC(=O)C(C)NC(=O)CCc1ccc(Cl)s1)NC(C1CCC1)=O Nc1nc(Cl)ccc1C(=O)NC1CC12CC(NC(C1CCC1n1cccn1)=O)C2 Cc1sccc1C(=O)NC(C(=O)N(C)CC1CC1)C1CCCO1 N1(C(CCCn2c(C)ncc2)=O)CC2CC1CN2C(=O)C=CC1CCCCCC1 C1(NC(C2(C)CC(C)C2)=O)CCCN(C(=O)Cc2cnn(C(C)(C)C)c2)C1C N1(C(C(C)(C)CF)=O)CCOCC(CNC(=O)C=CC(c2c[nH]cn2)=O)C1 c1(CCC(=O)NC(CCN(C(C=CC=CC)=O)C)C)ccc(F)c(OC)c1 C1(OCC(N2CCC(N(C(C3CCC(CC)O3)=O)C)C2)=O)CCC(CC)CC1 N1(C(CCC)=O)CCC(C(=O)NC(CN(C)C(C2OCCO2)=O)CC)C1 N1(C(C2(C)CC2)=O)CCCC(NC(=O)COc2c(F)cccc2Cl)C(F)C1 C(C(C)(C(=O)NOCC(N)=O)NC(=O)CC(C)NC(C)=O)SC c1(NC2CCCN(C(CC(C)C3CC3)=O)C2)ncnc2c1nnn2C1CC1 CC1(C)CCCN(C(c2cc(S(C)(=O)=O)co2)=O)C1CNC(C1CCSCC1)=O C1(C2CN(C(C3Cc4nnsc4S3)=O)C2)(NC(Cc2nnc(C)o2)=O)CC1 C1(C2CCCN(C(c3cnn(C)c3)=O)C2)(NC(C2=CCC(C)CC2)=O)CC1 C(=O)(C(F)(F)C(O)C1CC1)NCC(C(C)C)NC(C1CC2(CSC2)C1)=O C(CC1=CCN(c2ccnc(CO)n2)CC1)NC(C(C1CCOCC1)C)=O c1(CC(N2CC3CC(N4CC(F)C4)C2C3)=O)cc(C(F)(F)F)ccc1F N1(C(CCC)=O)CCC(NC(=O)CCN2CCN(C)CC2)C(C)C1 C1(CNC(CCc2c(C)ncs2)=O)CCCCN(C(c2ccc(O)nc2)=O)C1 C1(NC(CCOCCN(C)C)=O)CCCCCC1NC(=O)C(F)(F)CO N1(C(c2c(C)[nH]cc2)=O)CCC2(CCCN(C(=O)C(C)NC=O)C2)CC1 CC1(C)OC2CC(C(=O)NC3CC(NC(c4cccnc4O)=O)C3)CC2O1 N1(C(C2C(C)(C)C2CNC(C2CC=CCC2)=O)=O)CCC(C2CCCC2)C1 c1(C(=O)NCC2CC(C)N(C(c3cncs3)=O)C2)nc2ccccc2nc1O N1(C(C2(NC(c3c(C)non3)=O)CC(O)C2)=O)CC(=O)N2CCCC2C1 N1(C(CC(C)n2cccn2)=O)CCOC2CCN(C(=O)C3=CCCC3)CC12 N1(C(c2cnn(CC)n2)C(=O)NC(C)C)CCOC(C(F)(F)F)(CC)C1 N#Cc1cn(CC(N2CCC(c3c[nH]c4nccc-4c3)CC2)=O)c(=O)nc1O C1(C(=O)NCC=CCNC(=O)CCn2ccnn2)CCC(C(F)(F)F)CC1 NC1C2CN(C(=O)NCCc3ccc(CSc4ccccc4)cc3)CC12 C(c1cc2ccccc2o1)=CC(N1CCN(C(C2C3COCC23)=O)C(CF)C1)=O c1(CC(C)C(=O)NCC2CC(NC(C3(F)CCCC3)=O)C2)cccc(Br)c1 C1(C(=O)NCC(C(=O)NCc2cc(CC)on2)N(C)C)CCCC(=O)CC1 c1(C(N(C(C2CC2CC)=O)CCCC)C)ccc(C(C)N)cc1.C(C)(C)NC(C)C c1(C(C)C(=O)NCC(C2CC2)NC(=O)C2=CCCC2)c(F)cccc1F c1(CN2CCCC(CNC(C(=O)OCC)=O)C2)cc(Cl)nc(Cl)c1 C1(C(C)(C)C)CC2(C(=O)NCC(F)(F)C3CCC3)COC1C2 c1(C(N2CC(C)(NC(C(CC)F)=O)C2)=O)ccc(N)cc1OC C1(O)(CC)CCC(NC(C2CCN(C(=O)CCC(C)(C)C)C2C)=O)CC1 CC1(C)COC(C(N2CCCCC(CNC(C3(CCF)CC3)=O)C2)=O)CO1 C1(NC(c2[nH]cc(CC)n2)=O)CCCC(NC(=O)CCn2ccc(C)n2)C1 c1(NCCCCS(C)=O)nc2ccccc2nc1NCc1ccc(Br)s1 CC1C(C)N(C)CCN1C(=O)CCCCN(C)C(C1CC(C2CC2)=NO1)=O O=C(N=c1ccn(C2CCOCC2)[nH]1)C1CCN(Cc2cc3ccccc3[nH]2)C1 C1(C(N2CCCC(CC(C)C)CC2)=O)C2CCN(C(C3(O)CCC3)=O)CC12 N1(C(C2CC=C(C)CC2)=O)CC2CCC1C2NC(=O)CCC(=O)c1ccncc1 C(c1c(Cl)nc2ccccn12)=CC(=O)NCCC(C)NC(CCCCOCC)=O C1(NC(C2CCCC2)=O)CN(C(=O)CNC2C(C)CCOC2)C2CCCC12 C=C(Cl)CC(C(=O)NC1CN(C)CC1O)NC(c1cnc(=N)[nH]c1)=O c1(OC)ccc(OC)c(COCOc2ccc(Br)cc2)c1Br c1(C(=O)NC2CC(NC(c3n(C)ncc3N)=O)C2)cc2ccncc2s1 N1(C(c2ncc(C)c(Cl)c2)=O)CCCN(C(=O)CCF)CC1c1ccccc1 C(CCC(=O)NC(C)(C)CNC(=O)Cc1csc(NC=O)n1)C1C(C)C1 Cc1cc(Cl)ccc1OC(C)C(=O)NCC(F)CNC(c1cnc2n1CCC2)=O c1(CC)ccc(C(=O)NCC2CC3(CC(NC(=O)CC4CC=CC4)C3)C2)c(C)c1 c1(CN(C(Cn2cc(CNC(CC=CCC)=O)nn2)=O)C2CC2)cccc(F)c1 C(=O)(CC(CC)CC)NC1C(C(N(CCC)C)=O)COC1 N1(C(CC2(CSC)CC2)=O)CCC2(CCCC(CNC(=O)C(O)C(C)C)O2)CC1 C1(C(N2C(c3cn(Cc4cccc(C)c4)nn3)CCC2)=O)CC2C(=O)CCNC12 C1(=CC(=O)N(C2CCN(C(=O)Cn3ccc(C(F)(F)F)n3)C2)CC)CCC(C)C1 CCCC(CNC(C1CC(N(C)C)C1)=O)C(=O)N1CCC(C)(CO)CC1.C(C)(=O)O N1(C(c2cc(OC)nc(C)c2)=O)CC(C2CN(C(c3cc(C4CC4)cs3)=O)C2)C1 c1(OC)cccc(OC)c1C(F)(F)F.c1(C(c2nnnn2C)N)conc1C(C)C C1(CNC(C(C(C)O)c2cccs2)=O)CN(C)C2(CCOCC2)C1.n12cc(nn1)C2 c1(C(=O)NCC2C(NC(C3C(C)C3)=O)CCCC2)ccc2c(c1)NC(=O)CN2 N1(C(C2(O)CCOCC2)=O)CCC(NS(=O)(=O)C(F)(F)F)C(F)C1.C1CN1 C(=O)(C(O)CCCNC(C1(C(C)(C)O)CC1)=O)NC(C(C)O)C Cc1cc(C(N2CCCC2C(C)NC(c2ccsc2C)=O)=O)no1 O=C(CC1=CCCCC1)NCCCC1CCCN1C(C1CNC(=O)C1)=O C1(C(=O)NCC2(C(C)NC(CN3CCC(C)C3)=O)CC2)CC2(C1)CS(=O)(=O)C2 c12nn3c(c1C(=O)NC2)CCC3.c1(CC(=O)OC)cn(CCCOCC(C)C)nn1 c1(C(CC(=O)NCC(C)NC(c2ncc(OC)cn2)=O)O)ccc(Cl)c(Cl)c1 CC1(C)CC(C(=O)NCCC2CCCCO2)CN(C(=O)CN2CCOCC2=O)C1 C(=O)(CCCCF)N1CC(=CC(=O)NC2CC2NC(N)=O)C1 N1(C(C=CCN(C)CC)=O)CC=CC(C(N2CCC(C(N)=O)C2)=O)C1 C(=O)(CN=c1[nH]c(=NCCC(=O)NOCC(C)C)[nH]c2cccnc12)NC c1(CC)nc(CC(=O)NC2CCCC2CNC(=O)C(CC)n2ccnc2)cs1 N1(C(CCc2cc(C)no2)=O)CCC2CC2(C(N2CC(=O)N(C)C(=O)C2)=O)CC1 CCCCCCCC(=O)N(C1CN(C(c2ccsn2)=O)CC1(C)C)C N1(C(CCC(N)=O)=O)CC(NC(c2ncc[nH]c2=O)=O)CC(F)C1 C(=O)(CCC(CC)CCC)NC12CCCC(NC(CCCC)=O)(C1)C2 c1(C(=O)NC(C)C(CO)NC(=O)Cc2ccsc2)cc(Cl)cc2c1NCCC2 C1(NC(N(C)CC2CCN(C(=O)OC(C)(C)C)C2)=O)CN2CCCC1C2 c1(C(N2CCCC(CNC(=O)CCC3CC3)C2)=O)c(F)ccnc1F C(C)(C)(C(=O)N(CCCCCNC(=O)CCc1ccncn1)C)OCC C1(NC(C2(COC)CN(C(=O)CCN3CCCCC3)C2)=O)CCCN(C)C1 C1(C(=O)NCc2cccc(NC(C)=O)c2)CN(S(=O)(=O)N(C)C)CCO1 N1(C(c2c(CC=C)ocn2)=O)CCN(C(C2(C)CC2)=O)CC1CCOC CCC(C#N)(CC)C(=O)N1CC(CNC(C2CC(C3CC3)=NO2)=O)C(F)(CO)C1 Cc1ccc(C(N2CCSCC2C(N2CC(O)(C(F)F)C2)=O)=O)c(F)c1 c1(C(CCCCC2(C(=O)NC(=O)C(O)Cn3cncn3)CC2)C)ccc(F)cc1 C1(C(=O)NC2(CNC(C3C(C)(C(F)(F)F)C3)=O)CC2)CC2(CCO2)C1 C1(C)(CCNC(c2ccc(OC)o2)=O)CCN(C(C2(C)CC=CCO2)=O)C1 c1(C(=O)NC2C(CNC(c3cc(CC)[nH]n3)=O)C2)cnccc1C(C)(C)C c1(CC)cc(NC(C2CC(NC(c3cn(C)cn3)=O)C23CCC3)=O)cc(C)c1 C12(C(N3CC(O)(CNC(C(C)NS(CC)(=O)=O)=O)C3)=O)CCCC(=O)N1CCC2 CCC(C(F)(F)F)NC(=O)COC1(C)CN(C(=O)CC(C)OC)C1 N1(C(CC(CC)SC)=O)Cc2ccnn2CC(NC(C2(CN(C)C)CC2)=O)C1 CC(C)C(O)C(C)C(=O)NC1CN(C(c2cccc3nsnc23)=O)CC1N=[N+]=[N-] C1(CNC(C=C(C)Cl)=O)CC2(CCC2)CN1C(=O)CNc1cc(F)cc(F)c1 N1(C(c2cnc(NCC)nc2)=O)CCC(CNC(c2cc(F)n[nH]2)=O)C(C)C1 CC(C)C(CC(=O)NCCCN1CC=CC1)NC(=O)CCOC1CCCC1 N1(C(CSCC#C)=O)CCC(C)(NC(c2cc(-c3ccn(C)n3)on2)=O)C1 C1(N(C(=O)C(CC(=C)C)CC#C)CCC(=O)OC)CNC(=O)C12CC2 O=C(CC1C(=O)Nc2ccccc21)NC1CCCC(Nc2ncncc2I)C1 c1(SC)ncc(N)c(C(=O)NCC2CCCCN(C(=O)C(C)(C)CN(C)C)C2)n1 CC(=O)CCCC(=O)NC1CC2C1CCN2C(=O)C(C)Oc1cccc(C#N)c1 N1(C(C2C3C=CSC23)=O)CCC2(CCCC2N2CC(F)(F)C2)CC1 c1(C(C)CC(=O)N(C2CC(NC(C3CC(F)C3)=O)C2)C)c(F)cccc1F CC(C)CC(C)(O)C(=O)N1CCC(CCNC(c2cc(C3(C)CC3)n[nH]2)=O)CC1 N1(C(CC2(CCC#C)OCCO2)=O)CCC(CNC(C2(C)CC3CC3C2)=O)CC1 c1(C(=O)NC2C(C)CCN(C(=O)CCC(C)(C)C)C2)ccc2c(c1)N(C)CCO2 CC1CCC(=CC(=O)NCCC2(C)CCN(C(C3(CO)CCC3)=O)C2)CC1 c1(CN2CCN(C(CNC(C3(C)CC(=C)C3)=O)=O)CC2)c[nH]c2cc(F)ccc12 C1(C(=O)OC(C)C)CCC(C(F)(F)F)N(C)C1.c1(C2C(=O)N2)ccc(O)cc1 O=[N+]([O-])c1cnc2cc(Br)ccc2c1-n1cc(C2(O)CC2)nn1.N1CCNC(=O)C1 C1(NC(CSCC(C)C)=O)CCN(C(c2nn(C(F)F)cc2Cl)=O)CC1C N1(C(C2C(NC(C=CC=CC)=O)COC2)=O)CCC(C)CC1C c1(C(=O)NC2CN(C(C3(C)CC(OCC)(OC)C3)=O)C2)ccc2c(c1)C(=O)OC2 Cc1ccc(-c2ccc(C(=O)NCCCCNC(=O)CCCn3ccnn3)s2)o1 Cc1cnc2c(C(N3CC(=C(F)CNC(C4CC4C#N)=O)C3)=O)cccn12 CC(C)(C)C(CO)C(=O)NCC1CCCN1C(=O)Cc1csc(=N)[nH]1 C(CS(=O)(=O)CC(=O)NC(C(=O)NCC1CC1C(=O)OC)C1CCCO1)OC c1(C(N(C2C3CN(C(=O)CCCCC(N)=O)CC23)C)=O)cc2ncc(Br)cn2n1 n1(CC#C)cc(C(=O)N(C(C)CCNC(=O)CCN(C)C(=O)OCC)C)cn1 N1(C(c2cncc(Cl)c2)C(=O)NC(CC)(C)C)CCCOC(CN2CCCC2)C1 C1(NC(c2occ(C)c2)=O)CC2CCC(C1C)N2C(=O)CN(C1CC1)C(C)C CCCCCCC(=O)NCC1(NC(=O)CSC2CC2)CC(F)(F)C1 O=C(CC(O)(C(F)(F)F)c1nc2ccccc2s1)NCC1(O)CN(C(=O)CCF)C1 C=CCN=C(NCCC(C)(O)COc1ccccc1)N1CCC=C(c2ccco2)C1 CCC(CCC(=O)N(C)CCO)OCCC(c1ccncc1)(C)C.C(C)(=O)O N1(C(CCOC(C)C)=O)CC(C2CCN(C(=O)COc3ccccc3Cl)CC2)C1 Cc1ccn(CC(=O)NC2CN(C(=O)C(F)(F)c3ccccc3)CC2O)c(=O)c1 C1(CNC(CCC2CCN(C(CC=C(C)C)=O)C2)=O)NC(=O)NC1=O c1(C(=O)NCC2(C)N(C(C3(CC)CC3(F)F)=O)CCC2)cc(OC)c(N)c(C)c1 N1(CC#C)CCC(C(=O)NC2C3CN(C(C4CCCNC4=O)=O)CC23)CC1 c1(CC(N2C(CN(C(COCC)=O)C)COCC2)=O)cc(F)ccc1OC c1(C(=O)NC(C)CCNC(C2SCCCS2)=O)cccc(C2CC2)c1 CCCCCCCCCN1CCC(O)C(C(N2CCC(C)C(O)C2)=O)C1 C1(CCNC(c2cccc(CNC(C3CCCO3)=O)c2)=O)NC(=O)NC1=O C(c1cccnc1)=CC(=O)NCCN(C)C(C1C(Cc2nc(C)on2)C1(C)C)=O c1(-c2nnc(OCc3ccc(OCC)c(C#N)c3)n2C)ccc2ncc(C)n2c1 CC1CCN(C(C2C3CC4C(C3NC(c3cc(C(C)C)on3)=O)C24)=O)CCS1 S(=O)(=O)(c1ccc(OC)cc1)NC1CCN(Cc2cn(CCOC)nc2)C1 C1(CC(=O)NCCc2ccc(CNC(C(CC=C)C)=O)cc2)CC(=O)NC(=O)C1 N1(C(CN2C(=O)C(C)C(C)C2=O)=O)C2CCCC1CN(C(C1(CF)CC1)=O)CC2 O=C(C(F)C(F)(F)F)NCC1CN(C(c2ccccc2C2CCC2)=O)CC1O N1(C(c2ccc(C#C)cn2)=O)CCCC2CN(C(=O)C(F)C3CCC3)CC12 c1(OCC(=O)NC2CC2CNC(c2cccc(F)c2)=O)ccc(Cl)cc1 c1(C(=O)NC23CN(C(c4c(Br)c(C)n(C)n4)=O)C(C2)C3)ccc2nccn2c1 N1(C(C(CC)O)=O)CCC2(CC1)CC(NC(=O)CN(C)C(N)=O)C2 c1(C(=O)NC2C(C)N(C(c3cccn3C)=O)CC2)cc2c(Cl)nccc2o1 Cc1cnc(NC2CCC(F)(F)C(C)C2)c(S(=O)(=O)NCCCCS(C)(=O)=O)c1 Cc1ccc(C=CC(=O)NC2CCCCC2C(=O)NC2(CCO)CCCCC2)o1 c1(C(N(C2CN(C(=O)CCOCC3CCCO3)C2)C)=O)cc2cccc(Cl)c2o1 Cc1nn(CC(F)F)cc1C(N1CCC12CN(C(=O)CCC(C)C#N)C2)=O Cc1nc2ccc(C(=O)NC3CCN(C(=O)CCc4ccsc4Cl)CC3)cc2[nH]1 c1(-n2cc(CCC(C)O)nn2)cccc(NC(=O)C(C#N)C2CC2)c1 N1(C(c2cc(C(CC)C)no2)=O)CCN(C(=O)C(F)(F)c2cnccn2)C(C)C1 CCCCC(CNC(=O)CN(C1CC1)CC)NC(c1csc(C(F)(F)F)c1)=O CC(Cc1ccccc1)C(=O)NC1CCC(NC(=O)CCCN2CCCCC2)C1 c1(C(=O)NCC2(CNC(C(CCCC)CC)=O)CC2)ccc2c(c1)OC(C)(C)O2 CON=Cc1ccc(C(N2CCN(C(=O)C(C)(C)CO)CC2CC2CC2)=O)cc1 c1(C(=O)NC(CC)CNC(=O)C(n2cnc(C#N)n2)C)cccc2ccnn12 c1(C(N(C(c2ccccc2)CNC(C(C)OC)=O)C)=O)cnc(C)c(C)c1 Cn1cc(Cl)cc1C(=O)NCCC1(NC(=O)CC2CCC(F)(F)C2)CC1 N1(C(CCCc2scc(C)n2)=O)CCCCC1c1nc(=O)o[nH]1 C(CC(C(=O)N(C1CCOC(C)C1)C)NC(=O)C(O)Cn1cncn1)OC N1(C(c2c(C)cno2)=O)CC(CNC(=O)CCN(C)CCO)CC1(C)C c1(C(=O)NC2(CC=C)CN(C(=O)CCC3CC3)C2)cc(Cl)cn1C Cc1nc2c(C(=O)NCC(CO)NC(=O)Cc3cc(Cl)cc(Cl)c3)ccnc2[nH]1 CCC(CC(C)C)C(=O)NC1CN(C(c2cccc(OC(C)(C)C)n2)=O)C1 C=CC1CCN1C(=O)C=CCN(C(=O)Cc1ccsn1)C C1(O)(N(C(C(CCC)OC)=O)C)CCN(C(C2CCCN2C(C)=O)=O)CC1 C=Cc1cc(C(N2CC(NC(=O)CC(O)C(C)C)CC(F)C2)=O)cc(F)c1 C(CCCCC(=O)NC1C2CCC1N(C(=O)CC1CC1)C2)NC(=O)OC(C)(C)C N1(C(C2C(=C)C2)=O)CCC(COC)(NC(c2cccc(CSC)c2)=O)CC1 C1(NC(C(CC)(CC)CN)=O)CCCN(C2CCc3cscc32)C1 CC1CCCN1CC(=O)NCC(=O)N(CCC(F)(F)F)C1CCCCC1 c1(C(N2CCC(NC(c3ccc(C)cc3F)=O)CC2C)=O)sc2nccn2c1C c1(C(=O)NCC=CC(N2C(C)CC(C)(C)C2)=O)cnn2cccc2c1 C1(N(C(CSC(C)C)=O)C)CN(C(c2ccc(C(F)(F)F)o2)=O)CCC1C CCC(C)(C)C(O)C(=O)NC1C2CN(C(c3ccc(C)c(F)c3F)=O)CC12 C1(C(=O)NC2CN(C(CN(C)C3CC3)=O)CC2n2ccnn2)CC(C)(C)CN1C CON(C(=O)CN(C(=O)C(c1ccccc1)C)C(C)C)C1CCOCC1 C1(NC(c2cc(C(C)=O)oc2)=O)CC2CCC1(NC(=O)CCOC1CC1)C2 C1(NC(C(C)(C)NC(C2N(C)CCOC2)=O)=O)CCOC12CCCC2 N1(C(C=CC(=O)OCCCC)=O)CCN(Cc2sccc2C)CC1C1CCCC1 c1(CCOC)nc(=NC(C(C)NC(c2cc(C(F)F)ccn2)=O)C(C)C)s[nH]1 N1(C(CCC2CCC(=O)N2)=O)C2CCC1CC(F)(CNC(c1coc(Cl)c1)=O)C2 c1(CCC(=O)NCCCCNC(C2(C(F)(F)F)CCC2)=O)c[nH]c2ccccc12 N1(C(C(C)OCC(C)C)=O)CC2(Cc3ccccc3)CCC1C2.C12CC1NC2=O c1(NC(C2CCN2Cc2ccncc2Cl)=O)c(Br)cc(F)c(F)c1F Cc1ccc(F)cc1CC(=O)NCC1CN(C(=O)C(O)C(F)(F)F)CCCO1 n1(CC(=O)NCC2N(C(COCCOC)=O)CCC2C)ncc2ccccc12 N1(C(=O)NCCCOc2c(C)cccc2)CCc2c(F)cccc2C1.C(C(C)SC)N c1(C(N2C(C(C)NC(CCOC)=O)CCC2)=O)cnc2c(c1)NC(=O)CO2 C(=O)(CCCCCC(C)(C)C)NCC1CCC(CNC(C(C(C)C)C)=O)C1 c1(C(N2CCCN(C(c3c(C)[nH]nc3Cl)=O)C(C)C2)=O)ncn2cc(Cl)ccc12 C1(C(N2CCC(N(CCO)C(C3SC4C=CC3CC4)=O)C2)=O)CC2OC1C1CC21 c1(C(N2CC(OCC)C(CNC(=O)CC3CCC(=O)O3)C2)=O)c(C)ccnc1O C1(O)(C(=O)NC(C)CNC(c2cnn(CC3CC3)c2)=O)CCOC1(C)C C1(N(C)C)CCCN(C(c2ccc(N3CCCS3(=O)=O)cc2Cl)=O)CC1 Cc1cnccc1C(=O)NCC1CCC1NC(c1cncc(N(C)C)c1)=O C1(CNC(c2c(CC)n[nH]c2)=O)CN(C(C2CCCC23CC3)=O)CC1C c1(C(N2CCC(C(C)(C)NC(CSCC=C)=O)C2)=O)cc(C)nc(Cl)c1N c1(CNC(=O)CC2(NC(c3ccc(F)c(I)c3)=O)CCC2)cc(Br)cc(Br)c1F c1(C(C(=O)NCCn2cc(CCC3CCOC3)nn2)(F)F)nc2ccccc2[nH]1 C1(C(=O)NC2C(NC(Cc3n(C(C)C)cnn3)=O)C2)CCC=CCC1 C12(CC(=O)NCC3CCCCO3)CCC1CN(C(c1ccc(F)c(Br)c1)=O)C2 N1(C(C=C(C)Cl)=O)CC2ON=C(CNC(c3nccc4occc34)=O)C2C1 CCCCC(C(=O)NCCCCNC(=O)Cc1cccc(C)c1Cl)NC(N)=O N1(CC(C)C)CCCCC1C(=O)N(CC(O)CN(C)C(C1CCC(=O)N1C)=O)C C1(NC(=O)CCCCC2CC2)CCC2(CC1)CN(C(C1CC3CCC(C1)O3)=O)C2 Cc1ccc(C)c(OC(c2nc(NC(=O)NC)cs2)=O)c1.c1(O)ncc(O)cc1Cl c1(OC)ccc(CCN(C2CC2)CC2(CO)CCNCC2)cc1 C(=O)(CCCC(F)F)N(C)CC1CCCC1NC(=O)COCC(C)(C)C N1(C(COC(C)=O)=O)CCN(C(c2cc(O)cc(Cl)c2)=O)C(c2cccnc2)C1 C#CC1(C(=O)N(CC(F)Cl)C)CN(C(=O)CCc2nccn2C)C1 C1(COC)CC(Cn2cc(CC(C)C)nn2)N(C(=O)C(c2ccncc2)F)C1 C1(NC(C(CC)Oc2ccccc2F)=O)C2CC3CN(C(=O)CCCF)C1C3C2 c1(CNC(CN(C(=O)Cc2cn(C)nc2C)CCOC)=O)cc(C)cnc1F C1(COC)(CNC(C2CCSCC2)=O)CN(C(C2CC(n3cnnc3)C2)=O)C1 c1(C(=O)NCCN(CCC)C(C2(C)COC2)=O)c(C)cc(Cl)cc1C c1(OC)ccc(C(=O)NCC2(F)CCN(C(=O)CC3NC(=O)NC3=O)C2)nc1 C(C1CCN(C(=O)Cc2nc(=N)[nH][nH]2)CC1)=CC(=O)NCC(CC=C)(F)F c1(CC)ccc(C(=O)NCC2CC(C)(C)CN2C(C2CC(F)C2)=O)cc1[N+](=O)[O-] CCCC(C)(O)C(=O)N(C)CCN(C)C(c1cccc(F)c1NC(C)=O)=O C(=O)(CCCCC(F)(F)F)N1CCC(N2C(C)(C)CC2=O)CC1.C1(OC)CCCC1 C1(NC(=O)CCSc2ccccn2)CCN(C(c2cc3c([nH]2)CCC3)=O)CC1F C(CC(=O)NC1CCCN(C)C1)(C(F)(F)F)NC(COCC(=C)C)=O C(CN=c1[nH]c2c(c(=NCc3cncc(F)c3CC)[nH]1)COC2)NS(C)(=O)=O Cn1cc(CCNC(c2ccc3c(c2)CCC(=O)N3)=O)c2ccccc12 C1(CSC)(NN2CCC(C(C)(C)O)C2)CCSCC1 C1(NC(C(C)CCN(C)C)=O)CCCCCN(C(c2cc(=O)n(C)o2)=O)C1 c1(-c2cn(COC)nc2)cnc2c(C(=O)NC3CCC(O)C3)c[nH]c2c1 c1(NC(C2C(NC(c3cnc(C)nc3C)=O)C2)=O)c(Cl)cc(F)cc1Cl N1(C(C2C(C)CCO2)=O)CCCC1(C)C(=O)Nc1ccccc1 C(CCCCCC(=O)N1CCOC(C)(C)CC1)NC(C1C(CC)CCCC1)=O N1(C(c2cc(C(=O)OC)no2)=O)CCC(C)(CNC(=O)COCCC(C)C)CC1 C12(NC(CCCOCC=C)=O)CCCC1CN(C(c1cnn3ccn(C)c13)=O)C2 N1(C(C2CC(=C)C2)=O)CC2CCC1C(NC(c1c(Cl)c(C)nn1C)=O)C2 CC1Cc2ccc(Br)cc2CN1N1CCC(N2CCN(C)CC2)CC1 N1(C(c2cnc(=N)[nH]c2)=O)C2CCC1C1CC1(NC(c1coc(Cl)n1)=O)C2 C1(C)(C(=O)NCC2N(C(CCCCCSC)=O)CC(O)C2)CCC(F)(F)CC1 c1(OC)cc(C(=O)NC(C)(CNC(=O)C(F)n2ccnc2)C(C)C)cc(Cl)n1 c1(NCC(C(=O)NC)C)cc(=NCC2CCC3(CCCCC3)CC2)[nH]c(C)n1 N1(C(CC=C(C)C)=O)CCN(C(=O)C(C)n2cncn2)CC1c1ccccc1 c1(C(C(=O)OC)(C)NCC2CCCCC2N)ccc(F)cc1Cl C1(NC(CNC(=O)OCC)=O)CC12CCC(NC(c1ncc(C)cc1C)=O)CC2 C1(NC(c2ccc(CC)o2)=O)(CC)CCN(C(C2(C3CCCCO3)CC2)=O)CC1 N1(C(=O)Nc2scc(C(=O)Nc3ncc(Cl)cc3Br)n2)Cc2cccc(Br)c2C1 C(N=c1nc2ncn(C)c2c[nH]1)C1CC(C)OCC1.N12CCCC(O)(C1)CC2=O C1(C(=O)NCC(=C)CC)CN(Cc2cc(CC)on2)CCO1 c1(NC(=O)NC2CCOCC2N2CCCC2)c(Cl)cccc1Cl C1(C(C(=O)NCCC)N(CC(c2ccsc2)C)C)CCC2CC1C2(C)C C(c1ccc(F)cc1F)=CCCNC(C1CCN1CC1CC(=O)NC1=O)=O N1(C(C2CCC(=C)CC2)=O)CC2(CCCC2NC(c2ccc3cncn3c2)=O)C1 C1(NC(C(OC)OC)=O)CN(C(c2nc(C3CC3)cs2)=O)C2(CCCC2)C1 N1(C(Cc2cc(C)sc2)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC(CO)C1 C1(NC(Cc2cn(CC)nc2)=O)C2CC3C(C2)C13C(=O)CCN1CCNC1=O C(=O)(CCCCCn1cc(-c2ccc(Cl)nc2)nn1)NCC(C)(C)OC c1(C(=O)NC2C3(CN(C(C=COCC)=O)C3)CC2)c(C)[nH]c2ccc(F)cc12 c1(C(=O)Nc2cncc(C(F)(F)F)c2)nc(Br)c2n1CCCC2 c1(C(=O)NCCNC(C)C(N2CCNCC2)=O)cc(C(C)(C)C)ccc1C(C)(C)C c1(C(N2CC(N(C(c3nc(C(C)C)sc3)=O)C)C2)=O)csc(S(C)(=O)=O)c1 N1(C(CCc2onc(C)n2)=O)CCC(F)CC1C(=O)NCCCC1CCCO1 N1(C(Cn2nnc(C)n2)=O)CCN(C(C2CCC2)=O)CC1c1ccc(F)cc1 CCCN(OC)C(=O)C(CNC(C1CCCN(C)C1)=O)OC c1(-c2nc(-c3ccc(C)o3)nn2CCOC(C)C)cnnc2ccccc12 CCC(CC(=O)N1CCC(NC(=O)C(C)NC(C)=O)C(C)(C)C1)CC(F)(F)F C(C1NCCc2ccccc21)N(CC(=O)Nc1cccc(C)c1)CC C(CC(=O)N(C1CCC1O)C)(C(F)(F)F)NC(C(C)(C)OC)=O N1(C(c2c(C)cc(Br)o2)=O)CC2(C(=O)N(C)C)CCC1CC2 C=CC(C)(CCOC)C(=O)NC1C2CC1N(C(C1(C)C=CCC1)=O)C2 N(C(=NCC(=O)NC)N1CCC(F)C1)CCOCC CC(O)CC(=O)NC(c1ccccc1)C(=O)NCCCCn1ccnc1 N1(C(CCCOCCC)=O)CCN(C(c2coc(N(C)C)n2)=O)CC1C c1(C(=O)NCC(c2cccc(C)c2)NC(CC(C)SC)=O)ncc(Cl)cc1O C(=O)(CCNCCOCCOCCN(C(C(=O)OC)=O)C)OCC N#CC1CCC(C(N2CCC(C(CO)NC(=O)CCc3cn[nH]c3)CC2)=O)CC1 c1(CCNCCCOCCOCC)ccccc1I N1(C(C2CCN(C)C2)=O)CCN(C(c2csc(-c3ncc[nH]3)n2)=O)CC1C(F)F c1(C(N2CC3C(CNC(C4CC(OCC)C4)=O)(CC3)C2)=O)cccc2nccn12 CC(C)CN=C(NCC(=O)NCC1CCS(=O)(=O)C1)N1CCCC(C(F)(F)F)C1 c1(C(N2CCN(C(C3CCC(CO)CC3)=O)C(C3CC3)C2)=O)n[nH]c2c1COC2 c1(C(=O)NCCC2CCCCN2C(=O)COC2CCOC2)ccc(Cl)c(F)c1 C(=O)(CC(N)CC(=O)NC1CCC2CC1CN2)OCC Cc1cc(CC(=O)Nc2ccc(-n3cccc3)cc2)n(C)n1 c1(NC(=O)NCCCn2c(C)ncc2)cccc(NCC(F)(F)F)c1 c1(OC(C)C)ccc(C(=O)Nc2cccc(CC3CC(=O)NC3=O)c2)cn1 C(=O)(CCCCCC(C)O)NCCOCCNC(c1sc(CC)c(C)c1)=O N1(C(CN(C(CCOCC#C)=O)CC)=O)CCC(CC)CC1 n1(C(C)C)cc(CC(CC2CCC2)NC2CC2)nn1 c1(OCC)ccc2c(c1)CC(C(=O)NCCN(C(=O)C=C(C)C(C)C)CC)CO2 N1(C(C=CSC)=O)CCCC(NC(=O)Cc2ccc(-n3cnnn3)cc2)C1C C1(NC(c2ccc(SC(F)(F)F)cc2)=O)CN(C(C2(O)CCOCC2)=O)CC1O C1(C(=O)NCc2ccc(CO)o2)CCCCCN1C(c1n[nH]c2c1COC2)=O Cc1ccc(C(N2CCC(CNC(C3C(C#N)C3(C)C)=O)C2)=O)c(C(C)C)n1 C1(C(=O)NC2(C#N)CCN(C(c3cc(OC)n[nH]3)=O)C2)CS(=O)(=O)CC12CCC2 Cn1ccnc(N(CCCCCOC2CC2)CCO)c1=O c1(C2CCN(C(Cn3cc(CC(=O)O)nn3)=O)CC2)nc2ccccc2[nH]1 C(=O)(C1CCCc2nccn21)Nn1cc(C2CCCN(c3cc(C)ncn3)CC2)nn1 N1(C2(C(=O)NCCCN(C(=O)C=CCO)CCO)CCC2)CCOCC1 Cc1cc(C)c(C(=O)OC(C)(C)C)cn1.n12cc(Br)cc1OC2=O c1(C(=O)NC(C)CCNC(=O)CCCc2ccc(F)cc2)cc(F)c(F)cc1N C1(C(=O)OC(C2C(C(N3CC(N(C)C4CC4)C3)=O)C2(C)C)=O)CN(C)CCN1C C(=O)(CC(CC(C)C)NC(=O)CC1CC2(CC2)CO1)Nc1c(O)ncc(C)c1 c1(NC(C(CO)NC(C(CC)CCOC)=O)=O)ccc2c(c1)CCC2 c12cccc(c1)C(=O)N2.CC(CC1CCCO1)C(=O)NC1CN(C(=O)C2CC2)C1 C1(NC(Cc2ncc(CC)[nH]2)=O)CCN(C(=O)C(c2ccccc2F)(C)C)CC1C c1(CNC2C(C(=O)NC(C(=O)OCC)C)C2)cc(Br)ccc1C Cc1ccc(C)c(C(=O)NC2CCN(C(c3cc(Cl)ncc3Cl)=O)C(C)C2)c1 CC1(F)CCN(C(c2sc(Br)cc2Cl)C(=O)NC2CCOC2)C1 c1(C(N2C(CN(C(C(n3c(C)ccn3)C)=O)C)CCC2)=O)ccc(C(C)O)cc1 c1(C(=O)NC2CC(NC(c3ccnc(C)n3)=O)C(O)C2)c[nH]c2ccc(Cl)cc12 c1(C(=O)NCCC(CNC(C2(C(N)=O)CC2)=O)O)cccc(Br)c1N C1(CC(=O)NCC2(C)CC(NC(=O)C=CC3CCC3)C2)CCS(=O)(=O)CC1 N1(C(C2(COC)CC=CC2)=O)CC(N(C(=O)C(=CC2CCCC2)C)C)C(C)(C)C1 C12CCCC1NC(=O)C2.C(=O)(C(C)NC(=O)C(C)=C(C)C)N(CC)CC C1(CNC(COCCC#C)=O)(CO)CC12CCN(C(=O)CSC(F)F)CC2 Cc1csc(Cl)c1C(=O)NCC1(NC(c2ccnc(-c3cccnc3)n2)=O)CC1 N1(C(c2cc(=N)[nH]cc2)=O)CC(NC(=O)CCC2CCOC2)C2(CCCC2)C1 C(=O)(C1CCc2ccc(C)cc21)N(CCCNC(C1C(Cl)(C(=O)OCC)C1)=O)C C12(CNC(c3nn(CC)c(C)c3)=O)CCCC1CN(C(c1cnn(C)c1)=O)C2 C1(C(=O)NC(C)CCN2CCCC2)CCC(C2CC2)N1C(=O)CCC1CC1CO c1(C(=O)NCC(C2CCCC2)NC(C2C(COC)C2)=O)n[nH]c2c1COCC2 c1(Cn2cc(CNC(C(=O)Nc3ccccc3)=O)nn2)cncc(Cl)c1Cl C1(O)(CCNC(CC(CC)OC)=O)CCN(C(C2(CN(C)C)CC2)=O)CC1 N(C1CCCc2ccccc21)C(=O)Nc1c2nc(C)nn2ccc1 C(c1ccc2c(c1)OCO2)=CC(=O)NCC1CCN(C(c2scc(OC)c2)=O)C1 C1(CCC)CN(C(=O)CC(Cl)Cl)CC1C(=O)NCCC(=O)NC.C1(N)CC1 CN1CCN(C(=O)CC2(C)CCOC2)CC1C(=O)NCc1ccnc(O)c1 CCC(CCc1ccccc1)C(=O)NCC1CCN(C(C2(O)COC2)=O)C1 CC(C)C(C)N=c1[nH]c(=NCc2ccc(N(C)C)nc2)c2ncccc2[nH]1 c1(C(N2C3C(NC(CC=CCC)=O)CC(C3)C2)=O)cccc2c1NCCC2 C1(CCN(C(CSC)=O)C)CCN(C(=O)C(C)OCc2ccncc2)CC1 c1(OC)nc(C(N2CCC(N(C)C(c3c(F)cccc3F)=O)CC2)=O)ncc1F C1(C(=O)NC(CNC(C2(SCC)CC2)=O)Cc2ccccc2)CCC(C)(O)CC1 c1(OC)cc(C(=O)Nc2ccc(C(C)(C)C)cc2)ncc1-c1ccnnc1 C1(F)(COC)CCCN(C(=O)C(C)CN(C(=O)CCCOC(C)=O)C)C1 c1(CCC(=O)NCCN(C(Cc2cc(C)nn2C)=O)C)cc(Br)ccc1C Cc1noc(C)c1C=CC(N1CCN(C)CC1CNC(C1CC12CCCC2)=O)=O C1(C(=O)NC(CC)C(F)(F)F)CC(O)CCN1C(c1ccc(OC)cc1F)=O c1(C(=O)NCCC2(C)CCN(C(=O)C3=C(Cl)CC3)C2)cc(O)nc(C2CC2)n1 c1(C(=O)OC)cscc1NC(=O)C(Cc1cnc[nH]1)NC(=O)C(F)OC(F)(F)F N1(C(C2CCC(C)CC2)=O)CC2(CCCC2NC(c2cnc3ccnn3c2)=O)C1 C1(C(N2CCCC(C)(NC(c3ccon3)=O)C2)=O)Cc2cc(Br)ccc2O1 CC(CC(=O)N1CC2CC2(CNC(=O)CC2CSC2)C1)CC(C)(C)C Cc1nc(-c2nc[nH]n2)sc1C(N1CCOCC1CNC(=O)CC(C)(C)O)=O c1(C(=O)NCC(O)CNC(C2CCCN2C(c2ccco2)=O)=O)cccc(O)n1 Cc1cc(C(=O)NCC2CCC(NC(c3ccns3)=O)C2)ncc1C(N)=O c1(C(N(C)CC2CCN(C(c3cncc(CO)c3)=O)CC2)=O)c[nH]cc(Cl)c1=O C(=O)(CCCCCC(C)C)N.C12C(C)CN1N(CC=C)CCNC2=O.C(C)=O c1(OC)ccc(CC(=O)NC2CN(C(c3ccnn3C3CC3)=O)CC2C)c(C)c1 CC1CN(C(C2CCNC(=O)C2)=O)CCN1C(=O)CSCC(F)F N1(C(c2cc(CCCCC)[nH]n2)=O)CCOCC1CNC(=O)CCc1cnoc1 C(C)(C(C)C(=O)NCC(O)CCOC)NC(CC1(CC)CCC1)=O C1(CC#C)(C(N2CCCC2(C)CO)=O)CCN(C(c2csnc2Cl)=O)C1 Cc1nc(Cl)ccc1S(=O)(=O)N1CCCC1C(=O)NC(c1ccc(F)cc1)C1CC1 N1(C(c2cc(OC)cc(CC)c2)=O)C2COCC1CC(NC(c1ccon1)=O)C2 C1(C(=O)NC2CCCC(C)C2)CN(C(C2CCC3(CC3)C2)=O)CC12CCC2 CC1CC2(C(=O)NC3(CNC(c4c[nH]cc4Br)=O)CCOC3)CC12 N1(C(c2cccc(NC(=O)OCC)n2)=O)CCc2c(F)ccc(CO)c2C1 C(=O)(C(O)CC[S+](C)C)N1CCC(CN(C(C(c2ccccc2)C)=O)C)CC1 C=CCCC(C(=O)N1CC(=O)NCC1C)NC(c1ccncn1)=O c1(C(=O)NC2(C)CC(NC(c3cn(CCCC)nn3)=O)C2)ccc(C#N)s1 C(=O)(C(O)C(C)(C)C)N1C(C(C)NC(=O)CCc2ccc(C3CC3)cc2)CCC1 C1(CCC(=O)NC(C(C)(C)C)CO)CCCCN(C(=O)CC23CCCC2C3)C1 N1(C(CC(C(F)F)NC(C(COC)N(C)C)=O)=O)CCCC12CCOC2=O C1(CC(=O)O)CC2(CC2)CN1Cc1cccc(-c2n[nH]c(-c3ccccc3)n2)c1 CC(F)(F)CCCN=C(NCc1ccc(S(C)(=O)=O)s1)NCc1nc(CO)cs1 CCCCC(CNC(c1cc(C)sn1)=O)NC(C1CCC(C(=O)OC)C1)=O c1(CNC2CC(C)CN(Cc3cncnc3)C2)c(F)ccc(Br)c1Cl c1(OC)ccc(Cc2nnc(N(CC(F)(F)Br)C)n2-c2ccccc2Cl)cc1 C(=O)(CCC(=O)OC)NCC1(NC(c2cn(CC=C)nc2)=O)CCCC1 CC1CN(C(=O)Cc2ccc(O)nc2)CC1C(=O)NC1CCCCCC1 C(C(=O)N1CC(C)(C(=O)NC(C2(CO)CC2)C)C1)(C(C)C)OC c1(C(=O)NC2(C)CC(NC(C3CCN(S(C)(=O)=O)C3)=O)C2)cc(Cl)ncc1N n1(CC)c(C(=O)N(CC(C)C(=O)N2CC(c3nncn3C)C2)C)cnc1O C1(CNCC(C)O)CCN(C(C2CCCC2c2cnn(C)c2)=O)CC1 c1(NCCCC(C)(C)NC(CCCCOC)=O)cc(C(C)(C)C)nc(Cl)n1 Cc1ccc(C2CC2C(=O)NC2CC3CC(NC(=O)C4=CC(C)(C)C4)CC23)cc1C C1(CNC(C(CNC(C(F)=C(C)C)=O)O)=O)NC(=O)CC1(C)C N1(C(c2c(CNC(C3C(C)SCCC3)=O)cco2)=O)CCCC(C)CC1 c1(OCC)cc(C(=O)N(CC(C)N(C(=O)CC(C)C(F)F)C)C)oc(=O)c1 CC(CCCC(=O)N1CCCC(CCO)CC1)NC(=O)CN1CC(C)(C)C1 CC(C)CCC(C(=O)NCc1nn(C)cc1CSC)NC(C1CC1(C)C(F)F)=O C1(CNC(C2C(C)(C(C)C)C2)=O)CCCCN(C(=O)CCc2ccco2)C1 C1(C(=O)NCC2=C(C)CCC2)(CC)CCN(C(=O)C(C)OC)C1.CCOC C(=O)(CC(C(F)F)C(C)(C)C)NCC(CC(C)C)NC(c1ncc(OC)cn1)=O C(c1ccccc1)=CC(=O)NCCN(C(CC1C(CC)C1)=O)C C(=O)(CC1=CCCC1)N1CCC(CC(=O)N(C2CCSC2)C)C1 C(=O)(C(C(C)C)NC(c1c[nH]nc1CCNC(c1ccsn1)=O)=O)OC CCCCCCC(CC)C(=O)N(CCN(C)C(=O)C1CC1)Cc1n[nH]c(O)n1 c1(CC)ccc(NC(=O)CCC2CCC(NC(=O)CC(CC)C3CCC3)C2)cn1 C1(NC(C2(C)CCC(=O)N2)=O)CCCC(C(=O)NCCC2CC(O)C2)CC1 N1(C(C=CC)=O)CCN(C(=O)CC2CCCN(C(C)C)C2)CC1c1cn[nH]c1 c1(OC)ncc(Cl)c(N(C(C)CCNC(c2cnc(O)nc2O)=O)C)n1 C1(NC(C2C(c3n(C)ncc3)C2)=O)CCCN(c2cncc(Cl)n2)CC1 N1(C(c2c(CC)cc(Cl)cc2)=O)CCC2CCN(C(=O)C#CC3CC3)C2C1 C1(NC(CS(=O)(=O)NC)=O)CS(=O)(=O)C2CN(C(C3CCCN(CC)C3)=O)CC12 CCC(C)(C)C(=O)NC(CCC1CCC1)C(=O)N(CC1CCC1)CC1CC1 C(C)(CC(C)N=c1[nH]c2ccc(C(N)=O)cc2s1)NC(CCCCC(CC)C)=O Cc1sc(S(N)(=O)=O)cc1C(=O)NC1C2CN(C(C34CC(CN3C3CC3)C4)=O)CC12 N1(C(CSc2cccc(OC)c2)=O)CCN(C(C2CC(F)(F)C2)=O)C(C)C1 N1(C(C(CC)C#N)=O)CC(CNC(=O)C(=Cc2ccccn2)C)CC(C)(C)C1 c1(C(N(C(C)CNC(=O)CCC2CCCC2)C)=O)c[nH]c2ccccc2c1=O N1(C(C(CC#C)(C)C)=O)CC2CCC1CN2C(=O)Cc1ccc(F)cc1F C1(C(N(CC#C)CC)=O)CCN(C(C2CCC2(OC)OC)=O)C12CCC2 c1(C(N2C3C(CNC(C(CC)OC4CCCC4)=O)C(C3)C2)=O)ccnc(Cl)c1F c1(-c2c(CN(CCC)CCC3CCCC3)csc2)ccc2c(c1)CCO2.OC C(C(C)C(F)C(=O)N(C12CC(C1)C2)C)NC(C=Cc1ccc(C)o1)=O c1(C(c2nnnn2C2(C)CC2)NCCC(COC)OC)c(Cl)nc(Cl)n1C Cc1cc(C)c(C(=O)NC2CCCC2(C)CNC(c2c(C)csc2C)=O)o1 C1(C)(C(=O)NCC2OCCN(Cc3c(C(=O)OCC)scc3)C2)CCC(C)CC1 N(C(=NCCF)NCc1cccc(OC)c1OC)CC(N(C(C)C)CC)(C)C C(C1=NOC2CCCCC12)NC1CCCC(C=C)C1 C12(CNC(c3c(C)oc(Cl)n3)=O)CCCC1N(C(c1cncc(N)n1)=O)CCC2 c12ccc(cn1)c(=O)o2.Cc1cc(CNCC(N2CCC2C(=O)N(C)C)=O)cs1 Cc1cc(C(=O)NCC(C)(O)CNC(=O)CCn2c(C)ccc2C)sc1Cl c1(C(=O)NCCN(C(C2CC=CCC2C(F)(F)F)=O)CC)c(C)cccc1F c1(C(N(CC(CNC(CNC(=O)NC)=O)(C)C)C)=O)ccc2c(c1)C(C)C(C)O2 c1(C(=O)NC2CCN(C(C3(OC)CCOC3)=O)C2)cc2cnn(C)c2s1 c1(C(C)(C)C)ccc(-n2nc(-c3cncc(F)c3)nc2)cc1.C1(C2CC2)CCCCO1 c1(NC(=O)NC)cc(OC)ccc1CO.c1(C(=O)OCC)c[nH]nc1.C1(C)CC1 c1(CCN(C)C)cccc(C(=O)NCC2C3CN(C(c4ccc(F)o4)=O)CC23)c1 c1(C(=O)NC(CN(C(=O)Cc2cccc(Cl)c2)CC)C)c2c(nn1C)CCSC2 CCCCCCC(C)CC(=O)N1CCCC(NC(=O)C=CC(C)=O)C1 C#CCC(C)(C(=O)NC(C)CC(C)C(F)F)NC(c1ccnc(C)n1)=O N1(C(c2c(CC)onc2)=O)CCCC(N(C(=O)C(c2c(C)noc2C)C)C)CC1 CC1CCC(NC(=O)OC(C)(C)C)CN1C(=O)Cc1ccc(O)cc1 C12(C(=O)N(C(C)Cn3cc(CN4CC5CC5C4)nn3)C3CC3)CC=CC(C1)OC2 N1(C(C(C(C)C)OCC)=O)CCC(NC(c2cccc(=S)n2O)=O)C(CO)CC1 c1(C(=O)NCC#CCNC(CCS(N)(=O)=O)=O)c(C2CC2)nn2ccccc12 C1(C(C)SC)(NC(c2ccccc2F)C)CCCOC1 C(=O)(C(C)(F)C(=O)NCC(C)(O)CNC(c1ccc(COC)o1)=O)OCC c1(CNc2cc(N(C)C)ncn2)ccc(C(C)NC(C(C)C)=O)cc1 c1(C(CCC(C)CCS)c2n(CCSC)nnn2)ccc(F)c(OC)c1 N1(C(C2CCCC(NC(C3CC4CC(=O)C3O4)=O)C2)=O)CC23CCC2(COC3)C1 C1(=O)CN1.C(=O)(COCCF)N1C(C)CC1.C(COC)S.CCO c1(CC)ccc(C(N2CC(C(N)=O)(CNC(C3CC4CCC3O4)=O)C2)=O)nc1 c1(C(=O)NC(CC)CNC(=O)C(C)Cc2cccnc2)cc(N)nc(Br)c1 C=C(Cl)CCC(=O)N(C1CCC(NC(=O)CNC(c2cscn2)=O)CC1)C c1(OC)ccc(CCC(=O)NCC2C(O)CCN2S(=O)(=O)c2cn[nH]c2)cc1O c1(C(=O)NCC2(CNC(C3C(C(=O)OC)CC3)=O)CCC2)sccc1C N1(C(c2c(CC)occ2)=O)CC(NC(=O)C(N2CCSCC2)C)CC2(CCC2)C1 CC1CC(CO)CN(C(C2(C3CC3)CN(C(=O)C(=O)C(C)(C)C)C2)=O)C1 c1(C(=O)Nc2ccc(C)cc2F)cc2cc(F)cc(F)c2o1 C(=O)(C(C)C(O)C(C)C)N1C(CC)CN(C(=O)CSC(C)C)CC1 c1(CC)conc1C(=O)NOCC(=O)N(C1CC(C(C)(C)O)C1)C c1(CC(=O)NCC(C2CC2)NC(CC(C=C)C)=O)csc2ccccc12 N1(C(c2cc(C)[nH]c2C)=O)CC(CNC(=O)Cc2ccncc2Cl)CC1(C)C C#CC1(C(=O)NC2CCC(CC)C2)CN(C(c2coc(C)n2)=O)C1 c1(C(=O)NC2CCCN(C(CC=C)=O)C2)cc[nH]c2nccc1-2 C(=O)(C1=CCCC1C)NC(c1cccnc1)C=CCNC(c1c(C(C)C)cccc1)=O N1(CC)CCCC(C(=O)NC2CC3(C2)CC3NC(=O)C(c2ccc(F)cc2)F)C1 N#CCCCC(=O)NCCCCCCNC(C1OCCC1c1ccccc1)=O Cc1cc(C(=O)N(CC(C)N(C(=O)CCc2c(F)cccc2F)C)C)nc(C)n1 Cc1nnc(CNC(=O)CCNC(C2CC23CCC3)=O)o1.n12cc(nn1)C2 C(CC(=O)Nc1ccc2c(c1)CC2)(C(C)C)NC(C(CC)N(C)C)=O N1(C(C(C=C)(C)CC)=O)CC2CCC1CN2C(c1ccc2ccnn2c1)=O N1(C(c2cc(C)nc(O)c2)=O)CC(NC(=O)C(C)C(F)(F)F)CC12CCCCC2 C1(NC(c2c(C)coc2)=O)CC(C)N(C(=O)CC(C)n2ccnc2)C1 C(=O)(C(CC1CCCO1)NC(=O)NCC(c1cccs1)C)OC C(=O)(C(C(C)C)SC)NCCC(C)N(C(C(CC)n1nccc1C)=O)C c1(OCC(=O)N(C2CCN(C(=O)CCN3CCCC3)C2)C)cccnc1Cl c1(C(N(CC(C)NC(c2ccc(C#C)o2)=O)C)=O)ncc(OC)nc1OC c1(CNC2CC(COC)OCC2)c(C)sc2ccccc12 C#CCCCC(=O)N(C)CC1CCCN1C(=O)C(C)NC(c1ccco1)=O C1(CNC(C)=O)CC2(CCN(C(c3cccc(OCC4CC4)c3)=O)C2)CO1 CCCC(O)CC(=O)N1CCOCC(CNC(=O)Cc2cncnc2)C1 C1(C(=O)NCC2(F)CCCN(C(=O)C(Cl)=CCl)C2)CCCCC12CCC2 C1(CNC(C(N2C(=O)CCC2=O)C)=O)CC2(CCN(C(=O)C=CCF)CC2)CO1 c1(CC)ccc(C(N2CCC(CNC(C3CC3C3CC3)=O)CC2)=O)cc1Br C(CCC(C)(C)C(=O)N1CCCC(C)(O)C1)NC(C=C(C)C1CC1)=O N1(C(c2sccc2C)C(=O)NCC(=C)C)CCC(C2CCOCC2)(C(=O)OC)C1 C1(CC(=O)NCc2ccc(C(=O)NCC3CC3Cl)o2)CCSCC1 c1(CNC(c2cnc(SC)o2)=O)cccc(CNC(c2n[nH]cc2C)=O)c1 Cc1ccc(C#N)c(N2CCC(NC(C3(C(F)(F)F)CCCCC3)=O)C(O)C2)n1 c1(CC)sc(C(=O)NC2CCN(C(=O)COc3ccc(OC)cc3)C2C)cc1C CC1(C)CC2(CO1)CN(C(C1CC(NC(C3CC4C=CC3O4)=O)CCO1)=O)C2 N1(C(C(C)OCCCC)=O)C(C(=O)NCc2ccnn2CC)CCC1C N1(C(C2(COC)CCCC2)=O)CCC(N(C(=O)CSS(C)(=O)=O)C)CC1 Cc1ccc(Br)c(C)c1C(=O)OC(=O)CN1C(=O)SC(C)C1=O CC1CN(C(=O)OC(C)(C)C)CC1C(N1CC(NC(=O)C=C(Cl)Cl)C1)=O N(C(=NCCS(=O)c1ccccc1)NCC(c1ccccc1)(C)O)C(C(C)C)C c1(OCCC(C)N(CCC)C)cccc(-c2nc(=N)[nH][nH]2)c1 c1(N(C2CCSC2)CC(=O)NC(C)C(CO)SC)cc(CC)ncn1.CCO c1(OC)c[nH]c(C(=O)NC2CCCC(N(C)C(c3c[nH]c(C(N)=O)c3)=O)C2)cc1=O c1(OC)ccc(NC(C2C(O)CCN2C(c2cccc(O)n2)=O)=O)cc1I C(=O)(C(CC(N)=O)NC(=O)CCOC1COC1)NC(C1CCCC(C)C1)C N1(C(C2(CC)CC=CC2)=O)CCC(CNC(c2cscc2C(F)(F)F)=O)C(C)C1 N1(C(CSc2nc(C)[nH]n2)=O)CC(O)CC1CNC(=O)CN(CC(C)(C)C)C C(=O)(CCS(N)(=O)=O)NC1C(c2cn(CC)nc2)OCC1.C12(C)CC(C1)C(=O)N2 N1(c2nccc(OCCC)n2)CC(C)(C)CCC1CNC(=O)C(C)SC(F)(F)F C1(NC(C2CCN(CC)C2)=O)CN(C(C2(C(C)(C)CC)CC2)=O)CCC12CCC2 CC1(C(=O)NCC(F)CNC(C2CN(C(N)=O)C2)=O)CCC(F)(F)CC1 N1(C(C2CC(n3ccnc3)C2)=O)CCCC(NC(C2(O)CC2)=O)C1 C1(C(=O)NCCCCCCNC(=O)C(F)C2CCOC2)CCC2(CC1)CC2(F)F C12(CCNC(c3ccc(F)cc3F)CC)CCC(C1)C2(C)C c1(CNC(c2scc(C(N)=O)n2)=O)ccnc(OC2CCCC2)c1 c1(CNC(=O)NC2Cc3n(C)cnc3CC2)nc2ccc(Cl)cc2s1 c1(C(=O)NCC2C(NC(=O)CNC(=O)NC3CC3)C2)cc2cc(Cl)ccn2n1 C12(C(=O)NC(CCC3CC3)C(=O)NC3(C4CCCCO4)CC3)CCCC1OCC2 CC1CN(C(c2ccnc(C(F)(F)F)n2)=O)CC(C)N(C(=O)CC2(CO)CC2)C1 C1(C(=O)NC(CCN(C)C(C2COCC2(C)C)=O)c2cccs2)CCCC(C)(C)O1 C1(C(C)(C)O)(CNC(c2ccnnc2)=O)CN(C(=O)CSC(F)(F)F)C1 CN1C(=O)OCC1C(=O)NCC(C1CCN(C(=O)C2CC2)CC1)=O.C(C(C)(C)N)O C1(NC(=O)CSc2cccc[n+]2[O-])CN(C(c2cc(C3CC3)no2)=O)C2CC12 c1(CN(CCNC(c2c(C(C)C)nco2)=O)C2CC2)cccc(-c2ccncc2)c1 C1(C(N(C2CCC(NC(c3cc(Br)n(C)n3)=O)C2)C)=O)CC(=O)N(O)C1 c1(C(=O)NCC(=C)CCNC(C2CCC(C(N)=O)C2)=O)cc2cccc(Cl)c2s1 C(CC1c2ccccc2CCN1C(=O)CCSC(F)(F)F)NC(CCCCC)=O c1(C(N2CC(NC(C(C#C)(C)C)=O)CC23CCC3)=O)nccc2cccnc12 CC(C)(CCCNC(=O)CCCOC(C)(C)C)C(=O)NCC1(C)CC=CCC1 c1(C(=O)NCC(CN(C(CC(=O)NCC)=O)C)O)cccc2c1NCC2 C12(COC)CC(CNC(C3CC3C(N)=O)=O)(CN1C(C1CC13CC3)=O)C2 c1(C(=O)NCC(N2CCN(C(CS(CC)=O)=O)CC2)C(F)F)cccc(Cl)c1C CN1CCCCC1NC(C1CCC(CNC(=O)COc2ccccc2)CC1)=O c1(C(N(C2CCN(C(C3CC(Cl)(Cl)C3)=O)C2)CC)=O)occc1C N1(C(=O)CSC2CC2)C(C(=O)NC2CCN(C3CC3)CC2)CCC1C1CC1 C#CC1CCN(C(=O)CC2(O)CCN(C(c3cc(Cl)c(Cl)s3)=O)CC2)CC1 c1(C(=O)NCC(C(C)C)(C)NC(=O)COCC2CCCOC2)cc([N+](=O)[O-])n[nH]1 c1(C(=O)NC(CCN(C(CC(C=C)C)=O)C)C)c(CC)nc2ccccc2c1C C1(NC(C(C)OC)=O)CN(C(c2cnn(CC)c2C2CC2)=O)CC12CCOCC2 c1(C2C(N(CC(=O)NCCN3CCCC3)CC)C2)ccc(F)c(F)c1 C(=O)(C(CCNC(C1(C)CC2CC2C1)=O)OC)NCC(COC)(F)F c1(C(=O)NCCN(C(COC)=O)CC2CC2)ccc(C)c(-n2ccnc2)c1 c1(OCC(CN(S(=O)(=O)CCCC2CCCC2)CCO)O)ccc2ccccc2c1 c1(C(=O)NCC(C2CC2)NC(=O)C=CSc2nc[nH]n2)cc(Cl)c(O)c(Cl)c1 c1(CCC(=O)NCC2C3CN(C(c4c(=N)[nH]cnc4)=O)CC32)nnc(O)nc1O N1(C(C(C)C2CCCC2)=O)CC2(CC(NC(=O)C=CCN(C)C)CO2)C1 c1(C(=O)NC2(CC(N3C(C)(CC)CC3)=O)CCCCC2)ccc(N)cc1Cl c1(C(=O)NCCCN(C(c2c(C)cc(O)nc2)=O)C(C)C)sccc1S(N)(=O)=O c1(C(N2CC(NC(=O)Cn3cccn3)C(O)C2)=O)cc2cccnc2cn1 c1(C(N2CCC(CC=C)(NC(=O)CC3CC3)C2)=O)cccc2cc(O)ncc12 c1(N2CCC(N3CCC3)CC(C)(C)C2)nc2c(c(=NCCC(F)F)[nH]1)COCC2 C1(NC(=O)CCCc2ccc(CO)cc2)CCN(C(=O)C(O)C(F)F)C12CC2 C(c1nc(C)c(C)[nH]1)=CC(=O)Nc1cccc(NC(C(CC)OC)=O)c1 Cc1cc(C)n2nc(C(=O)NCC3CCN(C(c4ccn(C)c4)=O)CC3)nc2n1 C1(CNC(c2nc(CCC)oc2)=O)CC(F)(F)CN1C(=O)C=CCN1CCCC1 c1(OC)ccc(C(=O)NCCCN(C)C(c2c(C)ccnc2Cl)=O)cc1Cl C(=O)(C1c2n[nH]cc2CCN1C(=O)CCOC1CC1)OC c1(C(C)(C)C)ccc(C(N2C3CN(C(=O)NC4CCC4)CC32)=O)cc1 C1(NC(CN(C(c2cscc2C#N)=O)CC)=O)CC2OCCCC12 C(=O)(C1=C(F)CN(C(=O)CC2COCCO2)CC1)NC(CCCC=C)C CC1C(NC(=O)Cn2cc(Cl)cn2)CCCN1C(=O)C(F)CC1CC1 c1(COC)cccc(C(=O)NCCCCNC(C2(F)CCOCC2)=O)c1 N1(C(c2cccc(OC)c2)=O)CCCC(C)C1CNC(=O)CN1CCC(C)CC1 C(=O)(C(F)C1=CCCCC1)NC1CCC(NC(c2n(C)ncc2)=O)CC1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC(C)N(C(=O)CC2C(C)(C)C2(C)C)CC1 CCC(C(=O)N(C1CC(NC(c2ccccn2)=O)C1)C)NC(=O)CSC C(c1c(C)coc1C)=CC(=O)NCC1CC(CNC(C(CC)=CC)=O)C1 c1(C(N2CCN(C(C3=CCCC3C)=O)C(C3CC3)C2)=O)c(Cl)ccc(F)c1N CCCC(CC(=O)NC(C(F)F)C(C)(C)C)NC(=O)CN1CCC(C)C1 c1(NCC(C)OC)cc(S(=O)(=O)NC(c2cccnn2)C)ccc1C#N O=CN1CCOCC1C(=O)Nc1cccc(NC(c2ccc(Cl)o2)=O)c1 c1(C(=O)NCCOC2CCN(C(c3n(CC)ncn3)=O)C2)cc2ccccn2c1 N1(C(c2c(CC)cns2)=O)CCC(C)(C)C1CC(=O)N(CC)Cc1ccncc1 C1(C(=O)NC2CCC(CNC(c3c(OC)cccc3)=O)C2)CC(=O)NC1(C)C N1(C(CN(C(=O)C(=O)O)C)=O)CC2(CCN2C(c2ccccc2)=O)C1 C1(C(=O)NCC2(F)CCCN(C(c3cc(CO)on3)=O)C2)CCc2nc[nH]c2C1 N1(C(C(C)N2CCC2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C(C)C1 C1(NC(C(CC)NC(C)=O)=O)C2CCCN(C(c3cc(C)no3)=O)C2C1(C)C c1(N2CC(C(COC(=O)OCc3ccccc3)=O)C2)nnnn1Cc1ccccc1 C1(N(C)C)CN(C(=O)C=CC2CCCO2)CC12CC2 N1(C(CCc2cnc(C)s2)=O)CC2CCC1C(NC(C1CC3(CC3)CO1)=O)C2 c1(CNC(=O)Cn2cncn2)c[nH]nc1C1CCN(C(C2CC=CCO2)=O)C1 C1(NC(CCCOCC=C)=O)CCCC12CCCN(C(=O)COC(C)=O)C2 C1(CNC(=O)CC2CCN(C(=O)CCC3CC3(F)F)C2)CCC(CO)O1 c1(C(N2CCC(N(C(=O)Cn3nnc(C)n3)CC)C2)=O)cncc(C)n1 Cc1cc(C(N2CCC(NC(=O)C3=CCCC3)C(CO)CC2)=O)cn(C)c1=O Cc1oc(CNC(=O)Cn2ccnc2)nc1C(=O)NOCCn1ccnn1 c1(C(=O)NC(C2CN(C(=O)CCOC3CCOCC3)C2)C)ccnc2ncnn12 c1(C(=O)NC(CC=C)CNC(c2ccnnc2)=O)cnn(CC)c1CC c1(C(=O)NCC2CCC2C(=O)O)ccc2ncccc2c1Br c1(C(=O)NCCCCCNC(CC2CC(CC)C2)=O)cnn2ccn(C)c12 C1(C(=O)NCCC(CNC(C2CC2C2CC2)=O)OC)CCC=CCCC1 Cc1cccc(C(=O)NCC2CC(NC(C3CNC(=O)O3)=O)C(O)C2)c1 CC1CCCN(C(=O)C=CCF)C1CNc1ncc(Cl)c(O)n1 N1(C(C=CCCC(C)C)=O)C(C(=O)N(C2CCOC2)C)CC2CC12 C1(CNC(C2C(C=C)C2)=O)(OC2CCC2)CCN(C(c2csc(CCC)n2)=O)C1 Cc1cccc(C(C)NC(c2ccnc(CO)c2)=O)c1.c1(C=O)cncnc1C C1(C(=O)NC)C=CCN1C(c1[nH]ccc1CNC(=O)COc1cccnc1)=O N1(C(c2ccc(C(C)=O)o2)=O)CCC(CN(C(=O)CSCCC(C)C)CC)CC1 Cc1cc(C(=O)NC2CC(C(=O)NC3CCCC(CO)C3)C2(C)C)c(C)s1 C1(C(=O)NC(C(C)NC(c2cn(CCC)nn2)=O)C)CC2(C1)CC1(CC1)C2 C1(C(=O)NC(C(=O)OC)C2CC2)(NC(COCC(=C)C)=O)CCSC1 CC(CCO)N=c1nc2scnc2c(NCCc2cocn2)[nH]1 CCCC(CC)C(=O)N1CCC(CNC(C2CN(C3CCC3)C2)=O)(COC)CC1 C1(C(=O)NCC2(CNC(CCC(C)(C)C#N)=O)CCC2)CCc2ccccc2O1 c1(C(=O)NC2C=CCN(C(C(C)OCc3ccccc3)=O)C2)ccc(=O)n(C)c1 Cc1nc2ccc(-n3cc(C4CC(NC(=O)C(C(C)C)N(C)C)C4)nn3)cc2[nH]1 N1(C(C(C(C)C)O)=O)CCC2(CCN(C(=O)Cc3ncccn3)C2)C1 C1(C(N2CC(NC(Cn3c(C)cnc3)=O)C2)=O)CCN(C2CC2)C1=O O=C(C1=CCCCCC1)NC(C(=O)NC1(CC2CC2)CC1)C1CCC1 Cn1ccn2ncc(CNC(c3cn(CCF)cn3)=O)c12 C1(NC(=O)Cn2ccc3ccccc23)CCC2CN(C(=O)C3=CCSC3)CC2C1 c1(C(=O)NC2C(CNC(C(CC)Oc3ccccc3)=O)C2)cnc(O)cc1OC C1(N(C)C)CCC(C(=O)NC2CCC(NC(=O)CN3CCCC3=O)C2)CC1 C1(N(C(C(C)O)=O)C)CC12CCN(c1ncc(OC(C)C)cn1)CC2 c1(CNC(C2OCCN(C(c3cc(OCC)ncc3)=O)C2)=O)ccc(Cl)cc1C CC1=C(C(=O)NC(CNC(=O)Cn2cncn2)C(C)(C)C)CCS1(=O)=O C(=O)(C1=Cc2ccccc2C1)N1C(C)CC(CNC(c2ccccc2F)=O)CC1 CC(C)CCC(O)C(=O)N1CCC(CCC(=O)NC2CC(C)CC(C)C2)CC1 C1(C(N2CC3(CCN3C(C3CC4CCC3CC4)=O)C2)=O)(CF)CC2(CCC2)C1 CC(C)(C)C(C(=O)N1CCC1CNC(c1cccc(N)c1F)=O)N1CCCC1=O Cc1noc(C)c1CCC(N1CCC(F)(CNC(C2CCCC23CC3)=O)C1)=O C1(CNC(=O)CCc2ccoc2)CN(C(=O)CCc2ncc[nH]2)CCC12CCC2 c1(C(N2CCN(C(C(C(=O)OC)(C)C)=O)C3C2C3)=O)cc2cc(F)ccc2o1 C1(NC(C(CC)CC)=O)CC(C)CN(C(c2cnc(S)n2C)=O)C1 Cc1nc(=N)[nH]c(=NCC2CN(C(C3(C4CCC4)CCC3)=O)CC(C)(C)C2)[nH]1 c1(C(=O)NC2CN(C(c3cc(OC)ncc3)=O)CC(C)C2)cn2cccnc2n1 N1(C(=O)NCCCCC(=O)OC)CCCC(O)(CN(C)C)C1 C1(c2c(Cl)cc(OC)cc2Cl)NC(=S)N(C2CC2C)C2=C1C(=O)N(C)C2(C)C c1(C(=O)NCC(CNC(C2(NC(=O)NC)CCCC2)=O)C)noc2c1CCCC2 C1(CC#C)(C(=O)NCC(CNC(c2ncoc2C(C)C)=O)CO)CCOCC1 C1(CCCF)CCCC1(c1nnnn1CCCC1CC1)NCc1cccnc1Cl c1(C(N2CC(C3N(C(C=CCC)=O)CCC3)(O)C2)=O)ccc2nc(CO)[nH]c2c1 N1(C(C(=O)NCc2ccc(C3(C)CCO3)cc2)=O)CCCC(C2CC2CO)C1 N1(C(C=C=C(C)C)=O)CC(C(=O)NCc2nc(C)cs2)CC12CCC2 Cc1ccc(N)c(C(N2CC3(C2)CN(C(=O)C(O)P(C)(C)=O)C3)=O)c1 C1(C(=O)NCCc2coc(C)n2)(COC)CN(C(=O)CCc2cnc[nH]2)C1 O=C(CCC=CBr)NC1C=CCN(C(c2ccc(C(F)(F)F)nc2)=O)C1 CC1=C(C(=O)NCC2CC(F)(CNC(c3ccc(C4CC4)o3)=O)C2)CCCO1 C(=O)(C1=CCCC1(C)C)NC1(COC)CCN(C(c2cc(C)c(Br)o2)=O)C1 c1(CC(=O)NC2(COC)CCN(C(=O)Cn3cnnc3O)C2)cccc(C)c1Cl C(=O)(C1CCCc2sccc21)NC1(C)CCCN(C(c2csc(C)c2N)=O)C1 c1(C(N2CCCC(N(C(C(COC)OC)=O)C)C2)=O)cccc(C(=O)OC)c1C N1(C(C(CC)C2CCC(=O)N2)=O)CCN(C(=O)Cc2nnc(S)n2C)C(C)C1 CC1(C(=O)NCC=Cc2cccnc2)CCCN(c2nnc(C3CC3)o2)C1 CC(C(=O)N1CCN(C(=O)COc2ccsc2Cl)C(C(F)F)C1)C(C)(C)C C12(CNC(C3(OC)CC3)=O)CCCC1N(C(c1ccc3c(n1)CCC3)=O)CCC2 C(=O)(C(C)(CC)CC)N(CC(CC)NC(=O)CCC1CCCO1)CC C1(C2CCN(C(=O)CC3CC4C=CC3C4)CC2)(NC(CC(CC)CC)=O)CC1 C1(N(C)C(C2CCCCC2)=O)CN(C(=O)CCc2ccc(O)cc2)CC12CC2 S(=O)(=O)(c1ccccc1N)NC(C1CN(C)CC1c1ccc(F)cc1)=O C1(C(=O)NC(c2cncs2)C)CSCN1C(=O)COC1CCCC1 C=CCC(CC=C)C(=O)N1CCC(NC(C2CCC(C(N)=O)C2)=O)C12CC2 C(=O)(CCN(OC)C(=O)C1CCC2(CC2)C1)N(CC(C(=O)OC)C)C CC1CCCCC1(C)C(N1CCC(F)(C(=O)N(C)CC2(C)CCCO2)CC1)=O N1(C(c2c(C)con2)=O)CC2(CCN(C(=O)C(CC(C)C)N(C)C)CC2)CC1C N1(C(C(C)(F)F)=O)CCn2cc(C(=O)NCCOc3ccccn3)nc2C1 N1(C(c2c(CC)csc2)=O)CC2CCN(C(c3cccc(C)c3Cl)=O)C2C1 c1(-c2nc(CCC)nn2-c2cccc(C)c2)cc(SC2CCCCC2)nc(O)c1 N1(C(C2CC(=C)C2)=O)CCC2(CCC2CNC(c2cnn(CCO)c2C)=O)CC1 C(=O)(C(F)C(=O)N1CC(C(O)C(=O)NC2CCN(C)C2)C1)OCC c1(CC(=O)NCC2C(C)CCN(C(=O)C=CCO)C2)ccc2c(c1)NC(=O)C2 CCCCCC(C)NC(C1(CO)CCN(C(C2CNC(=O)N2)=O)C1)=O N1(Cc2ccc(OCC)cc2O)CC2CN(C(=O)CCC3CC3)CC2C1 C(=O)(C1=CC2(CCOC2)C1)NC(C1(O)CN(C(C(CSC)O)=O)C1)C c1(C(=O)NC2C(C)CN(C(=O)C(F)(F)C(F)(F)F)C2)ccc(F)c(S(N)(=O)=O)c1 c1(OC)ccccc1C(=O)NCc1cn(C2CCCC=C2Br)nn1 N1(C(C2(CC=C)CCOC2)=O)CC2CCC(C1)C2CNC(=O)CC1(OC)CC1 Cc1nc(=N)[nH]c(C)c1C(=O)NC(C1CCCCN1C(=O)CCOC(C)C)C CCC1=NOC(CC(=O)NC(C(=O)Nc2ccc(OCC)cc2)C2(C)CC2)C1 c1(C(N2C(C)(CNC(CCCC)=O)CCC2)=O)ccc(O)cc1O C(N=C(NC(C)C1CC1)NC1CC(OC(C)(C)C)C1)c1nc(CC)sc1 C1(CC(=O)NCCNC(=O)NCC)CC(C)(C)CN1C(C1C=C(C)CS1)=O c1(C(=O)NC2COCCN(C(CC(C=C)C)=O)C2)cc(N)c(O)c(F)c1 c1(N2CCCC(NC(=O)NC)C2)nc(=NC)[nH]c(=NC(C)C)[nH]1 c1(C(N2C(CC)C(NC(=O)CCc3cnc[nH]3)CC2)=O)cnc2n1CCC2 c1(C(=O)NCC2(OC)CN(C(C3CCCC(=O)N3)=O)C2)cc(Br)n(C)c1 N1(C(C2OCCC(C)C2)=O)CCN(C)CC1CNC(C1CC12CCC2)=O CC1CN(C(=O)N(C(C)(C)C)C(C2(F)C3CCCCC23)=O)c2cccnc2O1 N1(C(c2c[nH]c(=NC)o2)=O)CCC2C(C(=O)NCC3(CF)CCC3)C2C1 C(C(=O)CCc1ccccc1)(C(C)C)OC(c1c(C(C)C)n[nH]c1)=O N1(C(CCC(C)C)=O)CCCCC(CCC(N2CCOC(C(=O)N(C)C)C2)=O)C1 c1(C(=O)NCC(C)N(C(c2c(CC)nccn2)=O)CC)cccc(Cl)c1F C1(COC)CN(C(c2ocnc2C(C)C)=O)CCN1C(C1CC2C=CC1C2)=O C1(NC(COc2c(C)cccc2)=O)CCCCN(C(=O)CSS(C)(=O)=O)C1 N1(C(C2CC(C)OCC2)=O)C2CCC1CN(C(=O)CNc1ncccn1)CC2 N1(C(CCOC)=O)CCC(CO)(NC(c2cccnc2NCCN(C)C)=O)CC1 C(=O)(C(CCSC)NC(=O)OC(C)(C)C)NC1CC(NC(CC(=C)C)=O)C1 c1(C(=O)OC)cncc(C(=O)NC2CC(F)(CNC(=O)C(C)O)C2)c1C C(=O)(C(F)C(C)CNC(=O)CN(C)C(=O)C1CC1)NCCC(=O)NCC(C)C CCCCC(O)CC(=O)NC(C)(C)C(=O)NCC1(O)CC=CC1 CCC(C)(F)C(=O)NC1CN(C(c2ccc(C)s2)=O)CC1F Cc1ccccc1CC1(C(=O)NC2(C)CN(C(=O)CCn3cc(Cl)cn3)C2)CC1 N1(C(CC(C)F)=O)CCC(F)(CNC(c2cn(-c3ccccc3)cn2)=O)C1 C(CC(O)C(=O)NCCOCCCO)NC(c1c(C)cco1)=O CC1(C)CN(C(=O)C(C)(C)C(C)(F)F)CCC1NC(=O)Cn1nccn1 C#Cc1cnn(C)c1C(=O)NCC1CCC1NC(=O)C(CC1CCCC1)C(C)C Cc1nc(CC(=O)NC2CN(C(=O)C3CC3)CC2c2ccccc2F)[nH]c1C N1(C(C2(C)CCCO2)=O)CC(O)(C2(CNC(c3cncc(F)c3)=O)CC2)C1 N1(C(CNC(CC)=O)=O)CCCC(C2(NC(c3ccc(=O)n(CC)c3)=O)CC2)C1 c1(OC)ccn2c(C(=O)N(CC(C)NC(=O)CCC3CC3C)C)cnc2c1 N1(C(CCCc2ncc(C)o2)=O)CCN(C(=O)Cn2cccn2)C(C)CC1C c1(CN2CCOCC(C(=O)NC(C(=O)OCC)C)C2)ccc2nc(O)[nH]c2c1 CCC(C)(C)C(O)C(=O)NCC1(C)CCN(C(C2CC(C)OC(C)C2)=O)C1 C1(C)(SC)CCc2ccccc2O1.C1(C(=O)CC)CCCCC1CO C1(CC(=O)N(CCC(=O)NCc2c(OC)scc2)CC2CC2)CCCN(C)C1 Cn1ncc(S(C)(=O)=O)c1C(=O)NCc1ccc(F)cn1 c1(OC)ccc2[nH]c(=NCCC3(OC)CN(C(c4cc(O)ncn4)=O)C3)sc2c1 CC1(C)CC(NC(c2ccsn2)=O)CN1C(=O)CCc1ccccc1Br C1(NC(C=NOC)=O)CCC2(CC1)CCN(C(c1n[nH]c3ccc(Cl)cc13)=O)CC2 Cc1ccc(-n2nc(CO)nc2-c2cc(-c3ccccc3C(F)F)[nH]n2)cc1F C1(C(N2CCC(CCNC(CC3C(CC)C3)=O)CC2)=O)CN2CCC1CC2 N1(C(CN(C(=O)CC(C)(C)C)CC(C)C)=O)CC(C)(C)C2COCC12 c1(C(N2C(C)CCC(NC(=O)CS(C)(=O)=O)C2)=O)ccc([N+](=O)[O-])cn1 C1(N(C(Cc2c(C)cccn2)=O)C)CCC2CN(C(=O)Cc3ccco3)CC12 N1(C(c2c(CCC)nco2)=O)CCC(COC)(NC(C2CCCCC2O)=O)C1 C1(NC(c2c(O)cc(C)nn2)=O)CC2CC1CN(C(=O)CC1CCC1)C2 Cc1noc(C)c1C(N1CC2C(CNC(c3cnc(C4CCC4)o3)=O)C2C1)=O c1(OC)cc(C(N2CCC(C(=O)NCc3cccn3C)C(O)C2)=O)ccc1I N1(C(c2c(CCC)n(CC)nn2)=O)CCCCC(NC(=O)C=CC(=O)N(C)C)C1 c1(C(=O)NCCC(=O)NCCc2ccc(F)cn2)cccc(F)c1F CC1COc2c(C(=O)NCC(C)CNC(=O)C(c3ccc(Cl)s3)C)cccc21 N1(C(C(C2CCOC2)OC)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC(C)C1 C(=O)(C#CC1CCC1)NCC(CCNC(c1cncs1)=O)OC C(CCCCC(=O)NCC1(CF)CC1)N(C)C(c1nccc(C2CC2)n1)=O c1(OC)ncnc(C(=O)N(C2CN(C(=O)CCCn3cccc3)CC2F)C)c1F CC1CCOCC1C(=O)NC1CC(CCNC(C23CC(F)(C2)C3)=O)C1 C1(NC(c2c(CC)nn(C)c2)=O)CCN(C(c2nnn(CC)c2C)=O)C1(C)C N1(C(CCCCC)=O)CCC(C)(CNC(=O)C2=NNC(=O)C2)CC1 N1(C(CCN(CC)CC(=O)OC(C)(C)C)=O)CC2CC(NC(C34CCC3C4)=O)C1C2 Cc1ncc(C(=O)NCC(CNC(C2CC23CCCC3)=O)CO)c(C)n1 C12(C(N3CC(O)(CCC)C3)=O)COC(C1)C(NC(C1CCCCN1C)=O)C2 CON1CCC(CC(N2CC(CNC(C3(C)CCC(C)CC3)=O)C(O)C2)=O)CC1 CC(CC1CCCC1)C(=O)NC(C)(C(=O)NCCc1ccccn1)C1CCC1 C1(O)(C(=O)NC(C)CN(C(=O)C(O)C2CCC2)C)CCCC(C)(C)C1 C1(NC(c2cnn3ncn(C)c32)=O)CCC2CN(C(C3(N(C)C)CC3)=O)CCC2C1 C(N=c1cc(Cl)nc[nH]1)C1(O)CCCN(C(C23CCCN(CCC2)C3)=O)C1 N1(C(C(C)(CC2CCC2)OC)=O)CCC(C2CCN(C(=O)C(O)C(C)C)C2)CC1 C(=O)(CCS(N)(=O)=O)N1CC(NC(C(c2ccc(N)cn2)C)=O)C(C)C1 Nc1nc(C(=O)NCC2(NC(=O)Cc3ccccc3Cl)CCC2)ccc1O Cc1ccc(OCC(=O)NC2(CNC(=O)Cn3cc(C#N)cn3)CCOC2)cc1 CCCCC(C(=O)N1CC2(CCN2C(=O)CCC2C(=O)NN=C2C)C1)N(C)C C1(OC)CC(F)CN(C(=O)C(C2CC=CCC2)NC(c2ccc(O)cc2)=O)C1 c1(C(=O)NC(CCCCNC(C2CCC(C)CC2)=O)C)cnc(N(C)C)c(Cl)c1 c1(C(=O)NC(CCOC)CNC(=O)Cc2ncoc2C)cc(C)c(Cl)cc1F c1(OC(C)C(=O)NCC2(O)CN(C(=O)COC3CCOC3)C2)cc(F)cc(F)c1 N1(C(C)C)N=C(C(=O)N(C2CCCN(C(=O)COC3CCCC3)C2)C)CCC1=O c1(CC(=O)NC2CC(NC(C3(C)CNC(=O)C3)=O)C2)ccc2nn[nH]c2c1 CCC(C)C(CNC(C1(NC(c2csc(C)n2)=O)CC1C)=O)CO c1(SCC(Cc2ccccc2)NC(C(C)(C)NC(N)=O)=O)ccc(O)c(Cl)c1 Cc1ccc(NC(=O)NC(c2cnccn2)C2CCOC2)cc1OC(F)F Cn1nc(C(=O)NCC2CCCN(C(=O)C(O)Cn3cncn3)C2)cc1O N1(C(C=C(C)Cl)=O)Cc2ccc(C(C)NC(=O)C(c3c(C)n[nH]c3C)C)cc2C1 c1(NC(N(C)C)=O)ccccc1CNC(=O)CNC1C(Sc2cscn2)CCC1 CC1CCOC1C(=O)NCc1csc(-c2cnn(C)c2)n1.C12CCC1CNC2=O O(NC(=O)C(C)(C)C1CCCN1C(=O)CCn1cnnn1)C(C(C)C)C c1(C(N2C(CCNC(c3ccc(C#N)cn3)=O)CCC2)=O)n[nH]c2c1COCC2 c1(COC(c2c(OC(C)C)nccc2)=O)nc2ccccc2[nH]1 Cc1cnc(C(N2CCN(C(c3cccc(Cl)c3C(F)F)=O)CC2C)=O)cc1Cl CC1=C(F)CN(C(C2(CNC(=O)CCC3CC(C)C3)CCCO2)=O)CC1 C12(C(=O)NC3(CC=C)CCN(C(C4CC4C(F)(F)F)=O)C3)CCC(CC1)C2(C)C c1(C(=O)OCC)cc(NC(=O)C(N2CCC(C)C2)=O)cnc1Cl C1(C(=O)NCC(C)(F)CNC(=O)CCc2nc(=N)[nH][nH]2)(CC)CCCO1 N1(C(CC(C)(C)C#N)=O)CCC2(CCOC2)C(CNC(=O)CSC(=N)N)C1 C1(C(N(c2ncc(F)cn2)C)=O)C2CC(O)C(C2)N1C(C1CC1Cl)=O Cc1nc2c(NC(C3(C)CCCN3C(c3ccc(Cl)cc3C)=O)=O)cccc2s1 c1(CC(N2CC(N(C)C(c3cc(Cl)cnn3)=O)C2)=O)cccc(F)c1F C(=O)(C#CC1CCCOC1)N1CCC(n2cc(C(CC)O)nn2)C1 N1(C(c2ccc(CC)[nH]2)=O)CCN(C(c2ncccc2COC)=O)CC1C c1(C(C(N2C(CNC(C(C)=C(CC)C)=O)C=CC2)=O)C)ccc(OC)c(F)c1 c1(OC)ncccc1C(=O)NC1CCC1CNC(=O)CC(C)n1ccnc1 c1(C(=O)NCC2CCC(NC(C3(Cl)CC34CCC4)=O)CC2)cncc2ccccc12 C1(NC(c2nncs2)=O)CC2CN(C(=O)CNC(c3ccco3)=O)CC12 c1(C(=O)NCCNC(C2CC(C#C)(O)C2)=O)cc(OC(F)(F)F)cc(Cl)c1 N#Cc1c[nH]cnc1=NCC1(C)CCC1.C(c1ccncc1)=CC(=O)N(C)C1CC1.CO c1(C(NC2CCN(C(=O)CS)C2)=O)cn(C(F)F)cn1.C(C)(C)SC S(=O)(=O)(c1cccnc1)N1C(C(=O)NC2CCC(F)(F)CC2)CCCC1 C1(CC(=O)NC2(CO)CN(C(C3(CCCC)CCCC3)=O)C2)CCC(C)(C)C1 Cn1ccc(C=CC(N2CCCC2CC(N2CCC(OC3CC3)CC2)=O)=O)c1 CCCCC(CC)C(=O)NC1COCC1CNC(C1CCC(N(C)C)C1)=O c1(CC)ccc(OC2CN(C(c3ccn(C)c3)=O)CC2(C)C)cc1Br c1(CC)c[nH]nc1C(=O)NCCOC1CN(C(c2cc(C)on2)=O)C1 N1(C(C(CC#C)NC(c2ccc(C#N)s2)=O)=O)CC(F)(C2CC2)C1 C1(CC(=O)NCC(C)N(C)C(c2cc(Cl)c(Cl)[nH]2)=O)CCCC(O)C1 c1(CC(=O)NC2CCCN(C(=O)CC3CC(=O)NC3=O)C2)cc(F)cc(Cl)c1 C(C)(C)(C(F)(F)F)OCC(=O)NC(C)CCNC(C1(F)CCCC1)=O N#Cc1ccccc1CCCNC(C1CCN1Cc1cnc(Cl)cn1)=O C1(CC(=O)NC2CCN(C(C3(CC#N)COC3)=O)CC2)CC2(CCCC2)CO1 C1(C(N2CC(NC(C=Cc3ccc(C)s3)=O)C(C)C2)=O)CC12CCCCCC2 C1(N(C)C(c2cnc(Cl)s2)=O)CN(C(C2CCCN(S(C)(=O)=O)C2)=O)CC1O c1(C(N2CCCS2(=O)=O)=O)ccc2c(c1)S(=O)(=O)N=C1CCCCCN21 C1(CNC(=O)CC2CCCCC2O)CCCCC1C(=O)NCC1C=CCCC1 c1(OC(C)C)ccc(=NC(=O)C(=O)NCC(C)(O)C2(C)CC2)[nH]n1 N1(C(CC2ON=C(C)C2)=O)CC2CN(C(=O)CCc3ccc(C)c(Cl)c3)CC2C1 N12CCC(O)(C1)C(F)(F)C2=O.C1(CC#C)(C(=O)NC)CCCNC1 C(CC(O)CC(=O)NCCC1CSCCN1C(c1ccc(F)c(C)c1)=O)SC N1(C(c2ccc(C)cc2Cl)=O)CC2CCN(C(C3CC4(C3)CC43CC3)=O)C2C1 C1(C(=O)NCC2C=CCC2)CNC(=O)CN1C(c1csc(Cl)c1)=O c1(CCC)occc1C(=O)NCC1CC1CNC(C1CCC(O)C1)=O C1(CC(=O)NC2CC(c3ccccc3)(OC)C2)CCOCC1(C)C C1(CNC(C(CCC)NC(C)=O)=O)CN(C(=O)CC2CC(F)(F)C2)CC(C)(C)O1 C1(C(c2ccccc2)=O)CC2CC1CO2.C12CCCN1C2=O N1(C(C2OCCN(CC)C2)=O)CCCCC(CNC(c2nnn(C)c2C)=O)C1 C=CC1CN(C(=O)C(F)CC(C)C)CC1NC(C1(CC2CC2)CC1)=O CCCC(C)(C)C(=O)N1CC(CC(=O)NCC(C)OCC)C2(CC2)C1 C1(C(N2C(C(C)NC(CC=C)=O)CCC2)=O)CCn2c(Br)cnc2C1 C1(CNC(c2ccc(C)cn2)=O)(CO)CC12CCN(C(C1CC1C)=O)CC2 C(C(C(C)(C)C)NC(C1CC=CCO1)=O)NC(CCc1onc(CC)n1)=O N1(C(CCCCCC)=O)CC2CC(NC(=O)CCC[N+](=O)[O-])CC2C1 c1(C(=O)NCC(C)N(C(=O)CCc2cnco2)C)cc(CO)n(C)n1 c1(N2CC(OC)(CNC(C3CCCC(C)C3)=O)C2)ccn2c(Br)cnc2n1 N1(C(C(C)OCOC)=O)CCC(C)(C)C1CNC(=O)Cn1cc(CO)nn1 C1(CNC(COCCCC(C)C)=O)CCCC2CN(C(c3ccn(C)n3)=O)CC12 C(=O)(C(C)(C)NC(=O)C(C)(C)C)NCC(=O)N(CCCCC)CCO c1(NCC2(N(CC)CC)CC=CC2)ccc(S(C)(=O)=O)cn1 C1(C(N2CC(NC(C3CC34CC(C)(C)C4)=O)C2)=O)(OC)CCS(=O)(=O)C1 c1(N2CC(O)(CCNC(C3(O)CCCC(C)(C)C3)=O)C2)nc(Cl)nc2c1CCC2 N1(C(C2(CC=C)CC2)=O)CCC(NC(c2ncccc2OC)=O)C(F)(F)CC1 C1(CCC(N2CC(Cn3cc(CCn4c(C)ncc4)nn3)C2)=O)CC(C)(C)CO1 N1(C(C(C)OCC=C)=O)CC2CCCC(C(=O)Nc3cc(F)c(F)cc3O)C2C1 c1(CC(C)C)ccc(C(=O)NCC(C)(C2CCC2)NC(c2csc(Cl)n2)=O)cn1 N1(C(N(CC(C)C)Cc2ccccc2)=O)CCC2(CCC(O)C2)C1 N1(C(c2ncn(C)c2)=O)CC(C2CCCN(C(=O)C(C)(C)C(F)(F)F)C2)C1 c1(OC)ccc2c(c1)CCC2NC(=O)NC1CCN(C(c2cccnc2)=O)CC1C N1(C(C(C(CC)C)OC)=O)CCC2CCN(C(=O)CSCC(C)=O)CC2C1 Cn1cc(Cl)c(C(=O)NCCCCCCNC(C2(C)CCCOC2)=O)n1 c1(C2CN(C(=O)NCC)C2)cc(C(=O)N(C)C)n(C)n1.c1(C(CN)O)cccs1 CC1(C)COC(CC(N2CC3C(NC(=O)Cn4ccccc4=O)C3C2)=O)CO1 CC1(C)C2CN(C(c3onc4ccccc34)=O)C(C(=O)NCC3(C)CC3)C12 c1(C(N(CCC(C)NC(C(C)SC)=O)C)=O)ccc2[nH]c(=N)sc2c1 c1(CNC(CNC(CC)=O)=O)ccccc1CNC(c1ccnc(C(F)(F)F)c1)=O N1(C(C)C(=O)Nc2cn(CC3C(CO)C3(C)C)nn2)CC(O)(c2cnn[nH]2)C1 c1(C(N2CCC2C2CCCOC2)CC)ncc(C)cc1Br c1(C(N(C)CCNC(=O)C(F)CC2CCCCC2)=O)c(S(N)(=O)=O)cnn1C c1(NC(C)=O)cnncc1C(=O)NCC(C(C)(C)C)NC(=O)CCCC1CCC1 c1(CN(CCCN(C(C(C)CC2CCCCC2)=O)C)C)ccc(Br)cc1Cl C1(NC(=O)C(O)CCn2cncn2)CCCC12CN(C(=O)Cc1csc(Cl)c1)C2 C1(C(=O)NCC2N(C(c3cc(C(C)=O)sc3C)=O)CCC2)CNC(=O)C(C)(C)C1 C(=O)(C(C)C(C)NC(C1(NC(c2ccc(=N)[nH]c2)=O)CC1)=O)OC c1(C(=O)OCC)cccnc1NCC1CCC(NC(=O)C(c2ccccc2)O)C1 C#CC1(O)CC(C(=O)NC2CC(C(=O)NC3(COC)CCOCC3)C2)C1 C(C(O)(CNC(c1ncc(C(F)F)s1)=O)CO)OC C(=O)(C(O)C(C)(C)C)N(C(C)C(=O)NCc1cnco1)CCC c1(CC(=O)N(C)CC2CN(C(=O)Cn3ncn(C)c3=O)C2)ccc2c(c1)OCO2 CC1CCN(C(=O)CCc2cnco2)C1C(=O)NCC1(C#N)CC1 c1(C(N2CC(NC(C3C(c4ccn(C)c4)C3)=O)C2)=O)cc2ccccc2oc1=O O=C(CC1CCCN1C(c1n[nH]c2cccnc12)=O)N=c1ccnc(F)[nH]1 c1(N(C)C)cncc(N(c2ccc(F)cc2)C(=O)N=S(C)S)n1 C1(NC(c2ccc(C)cn2)=O)CN(C(C2(C)COC2)=O)CC(F)(F)C1 C(C)(N=c1ccc2c([nH]1)CCCC2=O)C1CCN(C(C(C(=O)OC)(C)C)=O)CC1 C(c1ccc(S(=O)(=O)NC23CCC(CC2N)C3)cc1)=CC(=O)NC1CC1 c1(CC#N)ccccc1C(=O)NC1CC=CCC1C(=O)NCCC12CCCC1C2 N(C(=NCC(C)C)NC(c1c(F)cccc1Cl)C)CC(c1cccc(OC)c1)O N1(C(C23OCC(COC)(C2)C3)=O)CC2CC(C1)C2NC(=O)Cc1ccccc1 O=C(C(F)C1=CCCCC1)N1CC2C(CNC(C34CCCCN3CCC4)=O)C2C1 C1(NC(C2(C)CN(C(C=C(C)C)=O)C2)=O)CNC(=O)C12CC2 C(CC(=O)NC1(C(=O)N(CC(O)C2CCC2)CC)CCC1)SCCCC c1(C(=O)NC2C(NC(c3cc(OC)n(C)n3)=O)CC2)ccc2cccnc2n1 c1(CC)cc(N)ccc1C(N1CC(NC(C2(C)CCNC2=O)=O)C(CC)C1)=O c1(C(N2C(CNC(CC(C)OC)=O)CC(O)C2)=O)ccc2c(c1)C(=O)OC2(C)C C12(C(=O)NCC3(C(C)NC(c4ccc(COC)cc4)=O)CC3)CCCC1OCC2 Cc1nc(C2CC2)[nH]c1C(N1CC(CNC(=O)CC2CCC(F)(F)C2)C1)=O C=CCC(CC(F)F)C(=O)NC1C2CCN(C(C3C(C)(C)C3(F)F)=O)CC12 CC12CN(C(=O)CC3(C(F)F)CC3)CC1CN(C(=O)C(O)P(C)(C)=O)C2 N1(C(C(C#C)(C)C)=O)C2CCC1CC(NC(=O)CCNC(=O)Nc1ccsc1)C2 Cc1cc(Cl)c(Cc2ccc(OC(=O)C(C)NC3CCCC3)cc2)cc1C c1(CC(=O)NCC2C(C)(C)N(C(C3CCSC3)=O)CC2)cc(F)c(F)cc1F c1(NC(CCCC=C)C)ncc(Br)cc1S(N)(=O)=O C(=O)(CCCCC(N)=O)N(C)CC1(CNC(C2C(C)(COC)C2)=O)CC1 N1(C(CC2CC(C(=O)OC)C2)=O)CC2CC(C1)N(C(=O)CC1OCCC1(C)C)C2 C1(CC(=O)NC(C(=O)NCC(CC(C)C)NC(N)=O)C)CN2CCN1CC2 N1(CC)CCCCC1CNC(CNC(Cc1cn(Cc2nonc2C)nn1)=O)=O C(C(C)(C)CN=c1[nH]ccc(=NC2CCCC2OC)[nH]1)OC CC(C)C(C)(CNC(c1ccn(C(F)(F)F)n1)=O)NC(=O)CC1CCCOC1 c1(C(N2CC(C)N(C(c3cccc4nccn34)=O)CC2)=O)ccc2cc[nH]c2c1 N#Cc1ccc(C(N2CCCC2c2nc(C(=O)NC3CC3)cs2)=O)nc1 C1(C(N2C(C(C(=O)NC3(c4c(C)con4)CC3)(C)C)CCC2)=O)CCCCC1F C1(N(CCNC(N2C(C(C)O)CC2)=O)CC2CC2)CCCCC1 C(=O)(N1CCC(NC(C2CC(C(=O)OCC3CC3)C2)=O)O1)C1CC(CCC)C1 Cn1cc(C(=O)NC2CCOCC2NC(C2(C3CCCO3)CC2)=O)c(C2CC2)n1 c1(C(N(C2CCCN(C(=O)CSS(C)(=O)=O)C2)C)=O)cnc2[nH]cnc2c1 c1(CC)cncc(CN2CCN(c3cccc(NC(=O)NC)c3)CC2)c1 N1(C(C2C(C(=O)OCC)CC2)=O)CCC(n2cc(CCSC3CCC3)nn2)CC1 C(CCCCC(=O)NCCC1CC(NC(c2nocc2C2CC2)=O)C1)OC C1(C(C(CC=CC)CC)=O)(CN)COC2(CCC2)C1 c1(CC)cc(OCC(=O)NC2(CNC(c3c(C)noc3N)=O)CC2)ccc1Cl C1(C(=O)OC)(NC(c2n[nH]c(COC)c2C)=O)CCC12CCC2 N1(C(c2cn(CCNC(C(CC)SC)=O)nc2)=O)CC(O)C(O)C1C(=O)O N1(C(C2(C=C)CCCC2)=O)CCCC(F)(CNC(C2CS(=O)C2)=O)C1 Cc1ccc(SC2(C(N3CCOC(C(C)NC(=O)CC(F)F)C3)=O)CC2)cc1 C1(NC(CCC(=O)OCC)=O)CN(C(=O)Cc2nonc2C)C(C)(C)C1 C(=O)(CC(O)C1CCCC1)NCC(=CC(=O)N(C(CC)C1CC1)C)C C(=O)(C(O)(C(C)C)C(F)(F)F)N1CC(C2CN(C(c3c(C)[nH]cc3)=O)C2)C1 C12(CC(=O)N(C3CCN(C(=O)CCS(N)(=O)=O)C3)C)CCCN1CCC2 C1(NC(CCC(C)OC)=O)CC2(C1)CC(C(=O)NCC(=O)OC(C)C)C2 CC(N)CCC(=O)N1CCN(C(c2ccoc2C2CC2)=O)CC1 c1(C(N(CC(C)N(C(CCn2c(C)ncc2)=O)C)C)=O)cc(N(C)C)ccc1N C(=O)(C(O)CCCC)NCC1(F)CC(NC(CCCNC(=O)NCC#C)=O)C1 N1(C(C(CC(=C)C)C)=O)CC2CCOC2(CNC(c2cc(N)ccc2C)=O)C1 c1(NCC23C(C)OC(C)(CC2)CC3)ccc2nccnc2n1 c1(OC)ccc(SCC(N2CC3CC3(CNC(=O)CC3CCC3OC)C2)=O)cc1 c1(C(N2C(C(=O)Nc3cc(OC)cc(Br)n3)CCC2C)=O)cccc(C#N)c1Cl N1(C(c2cc(CC)cc(N)c2)=O)CC2CCC(C1)C(NC(C1CC1F)=O)C2 CC1(C(=O)NC2(c3cn(CCOC4COC4)nn3)CCOC2)CNC(=O)C1 C1(C)(C(=O)NC(CC)(C)COC)CCN(C(=O)C2=CCOCC2)CC1 N(C1COc2cc(Br)ccc21)CC(=O)Nc1nnc(C)n1C N1(C(Cn2nc(C)c(Cl)c2)=O)CC2CN(C(=O)CN(C)CCO)CC2C1 c1(NC(C)=O)ccc(N)c(C(N2CC(F)(F)CC2CCNC(=O)CC(C)C)=O)c1 C#Cc1ccc(C(=O)NCCC(C)NC(=O)C(C)(O)C2CCC2)nc1 C(CCC(O)C(=O)NC1CC(N2CCC2)C1)NC(c1c(C(C)C)c[nH]c1)=O CCC(CC)(CC)C(=O)NCC12CC1CN(C(=O)Cn1cnc(C(N)=O)n1)C2 C1(C(=O)NCCC2OCCC2C)(CC)CCN(C(c2coc(C(N)=O)c2)=O)C1 C1(CNC(C(=O)NCC(N(CC)OC)=O)=O)CCC2(CC1)NC(=O)N(C)C2=O c1(OC)cc(C(=O)NCCCOCCNC(C2CCS(=O)CC2)=O)nn1C CC1(C)CCC=C(C(=O)NC2CN(C(=O)CN3CCCNC3=O)CC2(C)C)C1 Cc1cnc(C(=O)N(C)CCN(C)C(c2cc(C3CCCCC3)[nH]n2)=O)nc1 c1(C(N2CCN(C(c3c(CC)scc3)=O)C3C2C3)=O)cc2ccncc2c(O)n1 C1(C(N2CCCC2C2CCN(Cc3ccc(Cl)cn3)C2)=O)CCCNC1=O c1(C(=O)NC2CN(C(c3cnc(CC)nc3)=O)C(C)CC2)c(F)cc(F)cc1Cl c1(C(=O)Nc2cn(CC)nc2)csc2c1CCN(C(c1cnc(Cl)cc1I)=O)C2 C(=O)(C1CCCn2cnnc21)NCCCN(C(C(CCC)NC(N)=O)=O)C c1(OC)ccc2nc(C(=O)O)ccc2c1O.C123CC(C1)(C(C)(C)O2)NC3 N1(C(C=C(CC)CC)=O)CCCC(N(C(=O)CCSC)CC)CC1 c1(C(=O)NC(CCOC)CNC(c2nn(C)cc2C)=O)ccc(N=[N+]=[N-])cc1 N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCC(O)C(C(=O)N(c2cccc(Cl)c2)CC)C1 c1(NC(C2CCCC2NCc2cnccc2Cl)=O)cccc(O)c1Cl C1(F)(C(=O)NCCOCC=C(C)C)CCN(C(=O)C(C)=C(C)C)C1 c1(C(=O)NC(COC(C)=O)C(N)=O)nnn(-c2ccccc2C)c1C c1(C(=O)NC2CN(C(C(CCC)OC)=O)CC2O)cc2c(nn1)OCCS2 c1ccc(F)c(N2C(=O)CNC2=O)c1.C1=CC(=O)NCCC1.CC(C)=CC=C C1(C(N2CCCC2)=O)CCCCN(C(C2CCCC2F)=O)C1 C1(F)(C(N2CCC(C(=O)NCC3CC3)C2)=O)CN(C(c2ccncc2)=O)C1 c1(CCNC(C2(c3cccc(C)c3C)CCC2)=O)c[nH]c2c(C)cccc12 c1(C(=O)NCC2C(CNC(c3csc(C(F)(F)F)n3)=O)C2)c[nH]c2cccc(F)c12 c1(NC(=O)NC(C)CCO)cc(Br)cc(Cl)c1F N1(C(C(C)(O)C2CCC2)=O)CCOC(CCNC(c2nocc2Br)=O)C1 CCC(c1ccccc1)=CC(=O)NCCC(C)(C)NC(=O)C=Cc1cc(C)no1 C12(C(C)(C)C)COC(C(N3CCC(C(CC(=O)Nc4ccsn4)C)CC3)=O)(C1)C2 c1(C(N2CC(F)(CNC(C(c3ccc(Cl)s3)C)=O)C2)=O)ccc(Cl)c(N)c1Cl c1(CC(=O)NCC(CC=C)NC(=O)CCC(=C)C)cn(C)c2ccccc12 c1(C(=O)NCCCC(C)(C)NC(Cn2ncn(C)c2=O)=O)ccc(C#N)c(Cl)c1 C1(C(=O)NC2(CC=C)CN(C(c3cc(O)ccc3OC)=O)C2)CC2CCC1CC2 c1(N2C3CC(CNC(Cn4cc(C)nc4)=O)CC2CC3)ncccc1S(C)(=O)=O CC(C(=O)NC1(C)CCN(C(c2cc(Cl)on2)=O)C1)C(C)S(C)(=O)=O c1(N(CC(C(=O)NC)C)C)nc2ncn(C)c2c(=NC(CC(F)(F)F)C2CC2)[nH]1 c1(OC)ccc(C(=O)NC2CCC(NC(C3CCC(F)(F)C3)=O)C2)c(C)c1OC CCN=c1[nH]c(C(=O)NCC(C)(C2CC2)NC(C2CCS(=O)(=O)N2)=O)cs1 N1(C(c2cc(C)c(Cl)s2)=O)CCCC12CCCN(C(=O)CCc1cnn[nH]1)C2 C1(C(=O)NC(C)(C)C2CC2)COCCN1C(=O)CCC(N)=O.N1(C(=O)NC)CCCC1 CC#CCC(C(=O)NCCC(C)C(F)(F)F)NC(=O)CCOC n1(CC(=C)C)nnnc1C(c1cnn(CCO)c1)NC(C)Cc1ccccn1 C(CCN=c1ccc(C#N)n[nH]1)(c1cccnc1)N(C)C C1(NC(c2c(OC)nsc2)=O)CCC(CC(=O)NCCc2cnccc2C)CC1 N1(CC#C)CCC(C(N2CC3CC2C3CNC(C2(COC)CCCO2)=O)=O)CC1 c1(CC#N)ccnc(N2CCN(c3cccc(C(=O)NCC4CC4)c3)CC2)n1 C1(CC(=O)NC(C#CC#C)(C)C)CCN(C(c2ccc(C(C)=O)o2)=O)C1(C)C C1(O)(C(=O)NC(C(NOC2CCCN(CC)C2)=O)C2CCC2)CCOC1(C)C c1(C(=O)NC(C#N)C(N)=O)cc(C2CC2)cc(F)c1.C12CCC(CC1)NC2 C(C)(CNC(C1CC(SC)C1)=O)(CC(C)C)NC(c1c(CC)occ1)=O Oc1cc(-c2ccc(N3CCCCC3)cc2)c2ccccc2n1 c1(CCC)cccc(C(=O)N(C)CCNC(c2cn(C(F)F)cn2)=O)c1 C(=O)(C(C)(C)C1CCCO1)NCC(C)(C)NC(=O)CNc1cnn(C(C)(C)C)c1 c1(C(N2CCC(C)C(F)(F)C2)C(=O)NC2CCOCC2)ccc([Si](C)(C)C)cc1 CCC(C(C)(C)O)NC(=O)CCN(C(C1CCC(SCC)CC1)=O)C(C)C N1(C(c2ccc(OCF)cc2)=O)CCN(C(=O)C(O)Cn2cncn2)CC1CO N1(C(c2csc3cncn23)=O)CCOC2(CCN(C(C34CSC(C3)C4)=O)CC2)C1 C1(CNC(C2(C)CCOCC2)=O)CC2CC1CN2C(c1cocn1)=O C(=O)(C(C)CC(N)=O)NC(c1cccc(C)c1)CNC(c1n(CC)ccn1)=O C1(C(=O)N)(C(CCNC(COC)=O)=O)CCCO1.C12(CC1)C(=O)NC2.C(C)(=O)OC.OC C1(CNC(CCN(C(=O)COC2CC2)CC=C)=O)CCCC1C CCC(C)(CO)C(=O)NC(CNC(=O)Cc1cc(OC)cc(F)c1)CC(C)C C(c1ccccc1F)=CC(=O)OC(c1ccc(C#N)cc1)C(C)C C1(CN(C=O)Cc2nccc(CC)c2)CCC2CCCC2O1 c1(NC(C2(NC(C(C)OC)=O)CC2(C)C)=O)ccc2c[nH]nc2c1 CC1CCC(CCNC(=O)NCCCn2cccn2)O1 C1(NC(c2c(OC)nccc2)=O)C(C)CCN(C(c2cnc[nH]2)=O)C1C C1(C(=O)NC2CCN(C(c3cnc(SC)n3C)=O)C2)CCn2ncnc2C1 C12(NC(c3cc(SC)oc3)=O)CCC(C1)OC2C.c12ncccc1CNC2=O C1(N=c2[nH]ccnc2F)(CCC)CCN(C(=O)C(C)Cn2ccnc2)CC1 c1(OC)ccc2[nH]c(C(N3CC4(NC(=O)C=C(C)Cl)CCC3CC4)=O)cc2n1 CC1CN(C(=O)C(F)(F)CCn2ccnn2)CC2(CCN(C(=O)C(C)(F)F)C2)O1 C(C(F)(F)CCC(=O)NC1CCCC(F)(F)C1)N(C)C N1(C(C=C(CC)C)=O)CC2CN(C(=O)CCc3ccc(F)c(OC)c3)CC2C1 N1(C(=O)CC=Cc2ccccc2)CCN(C(C2CC3CC(=O)C2O3)=O)C2(CC2)C1 c1(OC)ccc(C(=O)NCC2CC(NC(=O)CCc3cnc(C4CC4)o3)C2)cn1 C(=O)(C1c2ccccc2C2CC1C2)N1CC(O)CC(NC(CCC=C(C)C)=O)C1 N1(C(C(C)N(C(=O)Cn2nnn(C3CC3)c2=O)C2CC2)=O)CCC(C)C1(C)C C1(OC)CCCCC1NC(C1OCCC1NC(=O)CNS(C)(=O)=O)=O N1(C(CCC(C)OC)=O)CCN(C(c2c[nH]nc2F)=O)C(CCO)C1 N1(C(c2ncn(CC)n2)=O)CCOCC1CNC(C1CC1CCOC)=O C1(NC(C(CCSC)O)=O)CC2CC(C1)N(C(=O)C(c1ccc(Cl)cc1)=O)C2 C(=O)(C#CC1CCCO1)NC(c1ccccc1OC)CNC(C(C)=C(CC)C)=O c1(OC)cc(N2CCC(CCNC(=O)C(F)C(C)C)CC2)nc(C(F)(F)F)n1 c1(CC(C(=O)OC(c2nccs2)CC2CC2)NC(C)C)cccc(Cl)c1 c1(C(N2CCC(CN(C)C(C3(Cl)CC34CCC4)=O)C2)=O)cc2ccccc2s1 N1(C(=O)NC(COCC=C)C2CCC2)CCOCN1C(=O)OC(C)(C)C c1(C(=O)NC2C(NC(C(C=CC)O)=O)CCCC2)cc2c(F)cc(Br)cc2[nH]1 C(=O)(CC(F)(F)Cl)NCCN(C(=O)C(O)C1CN(C(=O)OC(C)(C)C)C1)CC c1(C(N2CCC(NC(C3(C)CC(=C)C3)=O)CC2C)=O)cccc2c1CCCC2 CC12CCC(C(N3CC4CN(C(=O)COCC5CCOC5)CC4C3)=O)(CC1)CO2 CC1(N2CCOCC2)CCC(NC(=O)Nc2ncc(C(C)(C)O)cn2)CC1 CC(CC(=O)NC1CCCC1CNC(c1cnco1)=O)C(C)(C)C O=S(=O)(c1ccc(=NCCc2cnoc2)[nH]c1)N1CCCCC1CC1CC1 CC(C)(CC(=O)N1CCC(C(F)CNC(C2CSC2)=O)CC1)C1CC1 C(=O)(C1Cc2ccccc21)N1CCC2(C(C(=O)NCC(C(CC)C)CO)C2)CC1 C1(C(=O)NCCC2CCN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)CC2(CC2)CO1 CCC(C)C(C(=O)NCC1CC1c1cccs1)NC(C1CC(F)(F)C1)=O C1(CCNC(C2CC3CC2C3)=O)CSCCN1C(=O)Cn1cc(C(F)(F)F)cn1 Cc1ccc(F)c(C(N2CCC(O)C(C(N3CC(C#N)C3)=O)C2)=O)c1Br c1(CC(N2CCOCC(CNC(c3cnc(S)[nH]3)=O)C2)=O)cc2ccccc2o1 C(CNC(c1ccc(C2CC2)o1)=O)(CC(C)C)NC(CCc1cnc(C)s1)=O Cc1ccc2nc(Cl)c(CN3CCCC3C(=O)Nc3ccc(F)nc3C)cc2c1 C1(C(=O)NC(C)C=CC(=O)N(CCCN=[N+]=[N-])C)CCCOCC1 c1(C(=O)NC2(CNC(C(C3CCCC3)OC)=O)CCCC2)cc(OC)cnc1F N1(C(Cc2n(C)ccn2)=O)CCC2CN(C(C3CCCS3(=O)=O)=O)CC12 C(=O)(CCP(C)(C)=O)N1C(C(=O)NCC2CCC(=O)O2)CC(OC)C1 N1(C(c2nn(C)c(Cl)c2)=O)CC2CN(C(C3CC34CCC4)=O)CC2(C)C1 N1(C(C(COC)COC)=O)C2CCCC1CC(NC(c1cc(Cl)cnn1)=O)C2 N1(C(c2cncc(NC)c2)=O)CCCC(O)(CN(C)C(C2CC(F)C(=O)N2)=O)C1 N1(C(CNC(CC(C)C)=O)=O)CC(NC(=O)C(C)C2CCCC2)C(C)(C)C1 C#Cc1ccccc1CC(=O)NC(C)C(C(C)C)NC(=O)C=CC(N)=O C1(O)(C(C(=O)NCCN(C(C(c2ccc(F)cc2)CC)=O)C)(F)F)CCCCC1 C1(NC(c2c(CC)n(CC)nc2)=O)CC2CC(C1)N(C(c1cc[nH]n1)=O)C2 C(CS(=O)(=O)CC(=O)NCC1(F)CCN(C(C2C3CC4C(C3=O)C24)=O)C1)OC Cc1ccc(F)c(CNC(C2(C)CC3C=CC2C3)=O)c1.c12cn(nn1)C2 C1(C(=O)NCC2(C(=O)Nc3cncc(Cl)c3)CCCO2)CCCC12CCC2 c1(C(=O)NC2C(NC(CCC3CCCN(C)C3)=O)C2)c(F)cc(F)cc1F C(CCC)(C(=O)N1CCOC(CCNC(=O)CCn2ccccc2=O)C1)=CCC N1(C(c2cc(C3(O)COC3)on2)=O)CC2CCN(C(C3SCCCS3)=O)C(C2)C1 N1(C(C2C(C)C2)=O)CCC(NC(=O)Nc2cc(Cl)n(C)n2)CC1 N1(Cc2c(OC)cc(Cl)cc2)CC2CC(NC(C3CC34CCOCC4)=O)CC1C2 Cc1nccc(S(=O)(=O)N2CCCC(C3CCCCN3C(=O)NC(C)(C)C)C2)c1Cl Cc1cncc(C(=O)N(C)Cc2ccccc2CNC(=O)COCP(C)(C)=O)c1 c1(C(=O)NCC(CNC(c2cncnc2C)=O)OC)cc2ccccc2c(=O)o1 n1(CC(=O)N(C2CCN(C(=O)C(c3ccnn3C)C)C2)CC)ccnc1C N1(C(C(N2C(=O)CCC2=O)C)=O)CCCN(C(=O)Cc2ccc(Cl)cc2)C(C)C1 C1(C(=O)NC(CC)CC)CC12CCN(C(C1(C)CC3(CCC3)C1)=O)CC2 C1(NC(C(C2CCOC2)N(C(CC)(C)C)CC(C)C)=O)CCCCC1 C1(C(=O)OC)CN(C(=O)C(=O)NCCCN(C)C)CC(C)O1 c1(-c2nc(C)c(NCc3ncn4ccccc34)cc2)c[nH]c2ncccc12 CC12CCOC(C(N3CC4(C3)CN(C(c3ccc(NC5CC5)nc3)=O)C4)=O)(C1)C2 c1(NC(C(c2ccc(F)cc2)N)=O)ccc2cnoc2c1 C1(C(N(C)CC2N(C(c3nccc(C)n3)=O)CCCC2)=O)CCn2cnnc2C1 c1(C(=O)NCC2CN(C(c3c(C)scn3)=O)CC2(F)CO)cc2c([nH]1)CCOC2 c1(C(N(C)CC2N(C(CC=CC=C)=O)CCOC2)=O)ccc(Cl)cc1O C1(CC)CCCN(C(c2cc[nH]c2)=O)C1C(=O)NCC(C)(C)C(C)O c1(C(=O)NCC(c2ccncc2)C)c[nH]nc1CCNC(c1cc(Cl)cs1)=O C1(CC(=O)NCC(C)(C)CNC(c2occc2F)=O)CCC12CCC2 Cc1ccc(NC(C2CC3(CC3)CN2CCCC2CCCC2)=O)cc1F Cc1cc(C(=O)NC2CCCC(NC(c3csc(C(N)=O)n3)=O)C2)nn1C1CC1 c1(OC)cnccc1C(N1CC(C)C1C(=O)NCCCC1(C)CC1)=O N1(CC)CCOC(C(N2CCC(C(=O)N(C)CC3(C)CCC3)(OC)C2)=O)C1 C1(NC(CC2(C)CCOC2)=O)C2CC1N(C(=O)C=C1CCCCC1)C2 C(=O)(CC1(CN(C)C)CC1)NC(C1CC1Cl)C N1(C(=O)OC)CCCC(OCCNC(c2cn(C)nc2CC(C)C)=O)C1 c1(CC)nnc2c(C(=O)N(Cc3cccnc3)CC3CC(C(F)(F)F)CO3)cccn12 c1(SC)ccccc1C(N1CC(NC(c2c(Cl)cnn2C)=O)C(SC)C1)=O C1(CNC(CCOCC#C)=O)CC2CN(C(c3ccccc3CC(C)C)=O)CC12 CN1CCCC(C(N2C(C(N3CCC(C)(O)C3)=O)CC3CC23)=O)C1 C(=O)(C1=NOC(C)C1C)N(CC(CC)NC(=O)CCCc1ncco1)C c1(CC#N)ccc(C(N2CCOCC2c2cn(CC3CC4CC4C3)nn2)=O)cc1 N1(C(CC(C)C(F)F)=O)C2CCC1CC(NC(=O)C(C)(F)C(C)(C)F)C2 C(=O)(C(O)P(C)(C)=O)NCC(C1CC1)NC(c1cn(C)nc1C1CC1)=O CC#CCCCC(=O)N1CCC(O)(CNC(c2cnn(-c3nccs3)c2)=O)C1 C(=O)(C(O)P(C)(C)=O)N1CCC(CCC)C1.C(CC(=O)NCC)OCC#C C1(C(N2CC(OC(F)F)C2)=O)CCNC1=O.C1(CC=O)CC(N)C1 C1(C(=O)NCC(CNC(c2ccn3c2CCC3)=O)O)CCCC(F)(F)C1 CCC(CC(=O)N(CC(C)NC(=O)C(CCOC)N(C)C)C)OC n1(CC(N2CC3C(C(=O)NC4CCNC4=O)C3C2)=O)nc(Cl)ccc1=O C(c1cc(OC)ns1)=CC(=O)N(CCNC(=O)CCc1cc(Cl)no1)CC C(=O)(C1CCc2c[nH]nc21)N(C)CC1OCCN(C(C2(C)CC(C)OCC2)=O)C1 Cc1ccccc1OC(c1nc(CNC(=O)CSCc2ccncc2)cs1)C C1(O)(CNC(CC2(NC(CCC3(C#N)CCC3)=O)CC2)=O)CC2CCC1O2 N1(CC(=O)NCC2CN(C(c3cncc(C4CC4)c3)=O)CCO2)CC(=O)NC1=O N1(C(C=C=C(C)C)=O)CCCC2(NC(=O)CCC(=O)N(C)C)CC2C1 S(=O)(=O)(CC(=O)N1CCC(NC(C2OCCCO2)=O)C1)NC N1(C(c2cccc(C)c2)=O)CC2CC1CN(C(=O)CCC1CNC(=O)N1)C2 C(C(CC(C)C)NC(C12CCC1CC2)=O)NC(c1nc(C)oc1)=O N1(C(=O)C=Cc2nccs2)CCC(=CCNC(C2(n3cncn3)CC2)=O)CC1 N1(C(c2ccc(C)o2)=O)CC2(C(=O)NCCC(F)(F)CO)CCC1CC2 Cc1nc2cncc(C(=O)N(C)CCN(C)C(C3CCCS3(=O)=O)=O)c2[nH]1 c1(CC(=O)NC(C2CCN(c3nnccc3C#N)CC2)C)ccc(S(C)=O)cc1 C(=O)(C(C)(C)CC1CC1)N1CCC(CN(C(CC2(CSC)CC2)=O)C)C1 N1(C(c2n(CC)nc(C)c2)=O)CCC2(CCCC2NC(=O)CS(=O)(=O)N(C)C)C1 N1(C(c2c(CNC(CNc3cn(C)nc3)=O)n[nH]c2)=O)CC2CC2(N)C1 N1(C(CC2CC(=C)C2)=O)CC2(CCN(C(c3ccc(CC(C)C)nc3)=O)C2)C1 c1(C(=O)NCC2CCC(NC(CCOC(C)C)=O)C2)ccc2c(c1)CCCS2 Cc1ccc(-c2ccsc2C(=O)O)cc1.C12(O)CCN(C1)C2 CN1CCCN(CCNC2CCN(C(=O)C(F)OC(C)(C)C)C2)CC1 N1(C(CC(=O)NCC)=O)CC2C(CNC(=O)CCC3CC3(Cl)Cl)OCC2C1 C1(C(N2C3C(CNC(C(C)CO)=O)(CCC3)CC2)=O)CCC2(CC1)CNC(=O)C2 C1(CNC(CC2(C(=O)OCC)CC2)=O)C(C)CCCN1C(c1occc1C)=O.COC C1(NC(c2cc(F)ncc2Br)=O)CN(C(=O)COc2ccsc2)CC2(CC2)C1 c1(C(=O)NC2CCC(N(C(=O)C=CC3CCCC3)C)C2)c(S(N)(=O)=O)cnn1C C1(C(=O)NCC(c2ccc(F)cc2)NC(C(COC)N(C)C)=O)CCN(C)CC1 N1(C(=O)C(O)CCNC(C2(F)CCOC2)=O)CCC2(CCO2)C1 C#CC(CC(C)C)NCc1cnn2c1OCC2 N1(C(C2(OC(C)C)CCC2)=O)CC2CC2(CNC(=O)CCCC2CC2)C1 Cc1cc(OC(C)C(=O)NCC2C(CNC(=O)CC3(CO)CCC3)C2(F)F)no1 C(c1ccccc1)=CC(=O)N(C1CCN(C(=O)C=C(Cl)Cl)C1)CCO c1(C(N(CCN(C(CC(CC)C2CC2)=O)CC)CC)=O)ncc(C)cc1F C1(C(=O)NC(C(C)NC(CN(C2CC2)CC)=O)C)CCC(O)CC1 C(=O)(C1CCCc2ncnn21)NCC1(NC(=O)CC(=O)NCCC2CC2)CCC1 CCC(CC(=O)NC(C)C(C)NC(c1nnn(C2CC2)c1C(F)F)=O)SC C(=O)(C1=CCCCO1)N1CCC(C(=O)NC2CC2c2ccsc2)(OC)C1 c1(-c2ccc(OC)c(OC)c2)ccc(C)n2cc(CN)nc12 c1(NCC(CNC(CC(CC(C)C)C)=O)O)cc2nn[nH]c2cc1[N+](=O)[O-] CC(C)CC(CNC(c1csc(CN(C)C)n1)=O)NC(c1ccccc1)=O C1(C(N(C)Cc2cnc(C)s2)=O)CC2(CCN1C(=O)CN1CC(CF)C1)CC2 C(c1cncn1C)=CC(=O)NCCCN(C(CC1C(C)OCC1)=O)C1CC1 C(CC)(CC)(CCNC(=O)C(C)(C)C(C)C)NC(CC1C(CC)C1)=O C1(C(N2CC3(CNC(C4(CO)CCCO4)=O)CC2CO3)=O)CC2CCCCN2C1 Cc1c(C(=O)NCC2(F)CC(C)C2)cccc1Cl.C1(C(=O)N)CC(=C2CC2)C1 C1(C(N2CC(N3CCN(C(C4C(C)CC(C)O4)=O)CC3)C2)=O)CCC(C)(C)OC1 Cc1ccc(CN2CCCC(C(N3CCCCC3CO)=O)C2)c([N+](=O)[O-])c1 C1(C(=O)OCC)CN(C(=O)NCc2cc(CC)ncc2Br)CC(C)(C)C1 C12(C(=O)NCC3C(CNC(=O)CC4CSCCS4)C3)CCOC1CCOC2 CCC(C)CC(C)N(C)C(c1cn(Cc2ccccc2)nc1-c1cncc(F)c1)=O C(C1=CCCN(C(=O)C(C)N(C)C)C1)NC(COCCC)=O C(=O)(C(O)C1=CCCCC1)N1CC(n2cc(-c3n(C)ccn3)nn2)C1 Cc1cc(C(N2CCN(Cc3cnc(Cl)cc3C)CC2)=O)cc(O)n1 Cc1nn(C)cc1C(=O)NCC1CCCC1NC(=O)C(c1cn(C)nc1C)C Cc1nc(C)c(CCC(=O)NCC(C)N(C)C(c2c(C)nnn2C)=O)c(O)n1 O=S(=O)(c1ccc(Br)s1)NC1CCN(Cc2csc(-c3ccc(Cl)cc3)n2)C1 N1(C(C=CCOC)=O)CCC(OC(C)(C)C)C1.c12conc1C(C)NC2=O N1(C(CC(C)(C)C)=O)CCCCC1C1CCCN1C(c1ccc2nnnn2n1)=O C=CC(CCC)CC(=O)N(CC(=O)NCc1ccccc1O)CCC c1(-c2n(C)ccc2)nc(-c2cncs2)nn1C1CCCSC1 Cc1csc(CN(C(=O)CC=CCNC(=O)C(O)CC2CCCC2)C)n1 Nc1cc(C(=O)NC2(C3CN(C(C4CCCSC4)=O)C3)CC2)c(F)c(F)c1F CCCCC(O)CC(=O)N(CCCCNC(C1(n2nccn2)CC1)=O)C C(=O)(C(C)S(=O)(=O)C(C)C)N(C1CC2N(C(CC(=O)NCC)=O)C(CC2)C1)C N1(C(=O)CC2COCCOC2)CCC2CCCC12C(N1CC2CC1C2)=O c1(CC(=O)NCC(c2ccc(OCF)cc2)NC(C(C)N(C)C)=O)cn(C)nc1Cl C(=O)(C1CCc2c[nH]nc21)NCC(C)CN(C)C(C1(Cc2ccccc2)CC1)=O N1(CC(N2CC(CC)N(C(c3nc(Cl)c(Cl)s3)=O)CC2)=O)C(=O)C(=O)N(C)C1=O C1(NC(c2c(OCCC)cccc2)=O)CCN(C(=O)CCOC(C)=O)CCC1CO CC(C)C(C(=O)NCC1CN(C(C23CC(C2)C3)=O)C1)c1cccc(Cl)c1 c1(CCCN(C)CC2CCCN2C(c2cnc(Cl)s2)=O)c[nH]c2ccccc12 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NC(C(C)NC(=O)COCC1CC1)C c1(CCNC(C(N2CCC(O)(C(=O)OC)CC2)=O)=O)cc2c(cc1O)OCO2 CC1CCCC(OCC(N2CCOC(CNC(=O)C(F)=CCCF)C2)=O)C1 C1(CCC(=O)NCC(=O)N(C2CCCOC2)CC=C)CCC(C(=O)OC)C1 C1(CNC(=O)CC2CCC3CC3C2)COCCN(C(C2(O)CCOC2)=O)C1 C(CCN=c1ccnc(NCCSCCO)[nH]1)c1ccc(C)cc1C C=C(C)CN=C(NCn1cc(CC2CCC2)nn1)N1CCC(COC)C1 C1(C(N(C)CC2(NC(C3CC3F)=O)CC2)=O)CCc2cc(Br)ccc2O1 CC1CN(C(C2CC(n3ccnn3)C2)=O)CCC1NC(c1ccnc(CO)c1)=O N1(C(C=CCC)=O)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1CC(=O)NC Cc1cc(F)cc(F)c1NC(N1CCCC(N2CCOC2=O)C1)=O N1(C(c2scc(OC)c2)=O)CC2CCCC12.C12(CCCO1)C(=O)NC2 C1(C)(C(=O)NC2(C)C(C)CCC2)CC(=O)N(C(C)(C)C)C1=O c1(C(=O)NC2CCN(C(c3c(C)nsc3)=O)CC2C)nc2cc(O)ccc2[nH]1 N1(C(CCSc2ccc(C)cc2)=O)CC(C2(NC(=O)CC3CCCCC3)CC2)C1 C(=O)(CCCC(F)(F)F)N1CCC(N(C=O)C)CC1.c1(C(C)C)cnc(C2CC2)o1 c1(C(=O)NCC(C)(C)CNC(c2cc(Cl)cnn2)=O)cccc2sncc12 c1(CC)ccc(C(=O)NCc2cc(C(N3CCC(C(F)(F)F)C3)=O)n(C)n2)cc1 C1(n2cc(C3C(OC)CN(C(=O)C(CCOC)OC)C3)nn2)C=CC(C)(C)CC1 C(=O)(C1=C(C#N)CCC1)NC(COC(C)C)C(=O)N1CCC(NC(N)=O)C1 c1(C(=O)NCCC(=O)OC2CCNCC2)ccc(C(F)(F)F)cc1 c1(CC)nc(NCC2C3CN(C(=O)CCCCN(C)C)CC23)c(C#N)cc1C C1(C2CCCO2)(C(N(CC(C)(C)CNC(c2cc3n(c2)CCC3)=O)C)=O)CCCO1 CCCCC(CC)CN=C(NCC1CCC1)N1CCN(c2cc(CC)sn2)CC1 c1(CC)cc(C(=O)N(CC(C)(C)CNC(C2(COC)CCCO2)=O)C)cc(O)n1 C(CC(C(=O)NCc1ncn(C(C)C)n1)NC(c1cccnn1)=O)OC C1(CC)CCN(C(=O)CCC(C)NC(c2cc(C)c[nH]2)=O)CC1 c1(OCCNC(C2(OC(c3c(C)cc(Br)o3)=O)CC2)=O)ccc(Cl)cc1Cl C1(C(=O)NCC2CCCN2C(c2ccccc2F)=O)CC12CCc1ccccc12 c1(C(C(=O)NCC=C)N(C)CC=C)ccc(C(=O)NC2CC2)cc1 c1(CC)nc(C)n(C)c1C(=O)NCC(CCOC)NC(c1cn(CC)cn1)=O Cn1ncc(C(=O)NC2CCCCC2NC(=O)Cc2ccnc(O)c2)c1N c1(C(N(C)CC2CCN(C(C(CC)OCC)=O)C2)=O)ccc(C(=O)OC)cc1 c1(OC)ncnc(C)c1C(=O)NCCCCCNC(c1c(C)cccc1Br)=O N1(C(c2c(OC)nc(C)cc2)=O)CCC2(CCC2)C(NC(c2snnc2C)=O)C1 N1(c2cc(N(C)CC3CC(O)C3)nc(COC)n2)CCC2(C1)OCCCO2 N1(C(C2(CC)CCCCO2)=O)C2CC1CN(C(=O)CC1CCC=CCC1)C2 c1(SCC)cccc(CC(=O)NCCC2(NC(C3CCN(OC)CC3)=O)CC2)c1 C(CC(=O)NCC1CN(C)CCO1)(C(F)(F)F)NC(C=Cc1ccc(C)cc1)=O Cc1cc(C(=O)NC2C=CC(C(=O)Nc3ncn(C)n3)C2)cc(C)c1 c1(N(C(c2c[nH]nc2CSC)=O)C(c2cnccn2)=O)cccc(C)c1.CCN CCCC(C)(CC)C(=O)NCC1CCN(CCc2cccc(C(F)(F)F)n2)C1 C1(NC(C2CCN(C(CC)=O)C2)=O)CC2(CCC(NC(=O)C(O)C(C)C)CC2)C1 C(C(=O)N1CC2(CCCO2)C1)(C(C)(C)C)NC(C(C)C#N)=O C1(C)(NC(C23CC(NC(C4C(C)CC(=O)CC4)=O)(C2)C3)=O)CN2CCC1CC2 c1(C(N(CCC)CCNC(c2cn(CCOC)nn2)=O)=O)ccc2scnc2c1 C(C1CCC(C)CC1)=C(C)C(=O)NCC(CC(C)C)NC(c1sc(C)cc1C)=O c1(C(=O)NCC2N(C(CC(c3ccc(F)cc3)C)=O)CCC2)ccc(C#N)cc1 C1(C(=O)NCC=COCC)CCCCC1(C)NC(=O)C(C1CCCC1)OC c1(NC(=O)NC(c2ncc[nH]2)C)ccnc(NC(C)(C)C)n1 c1(C(N(C2CCCN(C(C(C)=C3CC3)=O)CC2)C)=O)sc2nccn2c1C N1(C(C=C(C)C(F)F)=O)C2CCC1C(CNC(C1CCC(C)(O)CC1)=O)C2 Cc1csc(C(=O)NC2(CNC(=O)C(C3CCCCC3)O)CCOC2)c1Cl C(CNC(=O)C(N1CCNC1=O)C)(C(=O)NCCC(F)F)OC c1(OC)ccc(CCCN2CCC(C)C2CNC(=O)C(C)OC)cc1 C1(C(N2CCN(c3ccccc3)CC2)=O)CSCCN1Cc1ccc(O)cn1 C12(C(=O)NC34CC(NC(C5C(n6ncc(C)c6)C5)=O)(C3)C4)CCC(CC1)C2 C1(C)(CC(=O)N(CC(C)OC)CC)CCN(C(=O)C(O)CN2CCCC2)C1 C1(NC(C2(CCOC)CC2)=O)CCN(C(c2c(OC)n(C)nc2)=O)CC1O C(c1cccc(Cl)c1)=CC(=O)NCC(CN(C(=O)CC12CC(C1)C2)C)O Cc1nnc2cc(N3CC(F)(F)CC3(C)CNC(=O)C=Cc3cccs3)ncn12 n1(C(C)C)nccc1S(=O)(=O)NCC1CCC(=O)NC1C N1(C(C(CC)n2ccnc2)=O)CCC2CC(NC(=O)CO)CCC2C1 C(C(CC(C)C)NC(=O)CCCc1cnn[nH]1)NC(CCc1c(C)ncs1)=O c1(C(=O)NCC2C(NC(c3c(CC)occ3)=O)C2)coc2cc(F)cc(F)c12 C(=O)(CCCCC(F)F)N1C(CC)C(NC(c2cc(C(C)C)cc(F)c2)=O)CC1 C1(NC(C2C(OC)CCC2)=O)CC=CCC1C(=O)Nc1ccc(CCF)cc1 c1(C(=O)NC2C(CNC(C=CC(C)SC)=O)COC2)ccc(F)cc1 c1(CC(=O)NCC2C(NC(c3c(C)cccc3F)=O)C2)ccc2ncccc2c1 c1(CC)cc(C(=O)NCC2CC2NC(=O)CCNC(=O)NC)c(C)o1 N1(C(c2c(CC)c[nH]n2)=O)CC(NC(c2coc(Br)n2)=O)CC1(C)C C12(CCCS(=O)(=O)C1)CN2.c1(N(C)CC)cc(Cl)ncc1F CN1C(=O)CCC1CC(N1CCC(C2CCCCN2C(=O)C(C)(O)C2CC2)C1)=O C1(CNC(COCCSC)=O)(CNC(C2CCC(=O)O2)=O)CCOCC1 c1(OC)ncc(C(=O)NC2CCC2CNC(c2cscc2Cl)=O)cc1Cl c1(C(N2CC3C(NC(C(CC)(C)C(N)=O)=O)C3C2)=O)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)OC)ccc(NC(C(=O)OC)C(C)O)c(Cl)c1 C(=O)(CCCC(C)NC(c1c(C)nn(C)c1N)=O)NC(CCSC)C CCC(CC)C(=O)NCCOC1CN(C(=O)C(C)C(=O)OC(C)(C)C)C1 CCCC(C)CC(C(=O)NCc1nnn(C)n1)N1CC2CC(C)(C)C2C1 N1(C(C2(SC)CC2)=O)CCOC2(CCC(NC(=O)CCc3nccs3)CC2)C1 C(=O)(C(C(C)NC(c1cnc(=N)[nH]c1)=O)C(C)C)NCCc1cn(CC)nn1 C1(S(C)(=O)=O)(C(=O)NCC(CCC)NC(c2cc(CO)c(C)o2)=O)CCCC1 N1(C(C(C)NC(C2CCCC2)=O)=O)CCN(C(c2cnco2)=O)CC1C(F)(F)F CN1C2CCC1CC(=CC(=O)NCC1CN(C(=O)C=CI)CCO1)C2 c1(NC(C)=O)ccc(C(N2CCN(C(C3CC(O)CN3)=O)C3CC23)=O)c(C)c1 c1(CCC)nn(C)c(OC)c1NCc1c(C)nn(C)c1C.c1(C(C)N)ccc(OC)cc1 Cc1c(Br)cc(C(=O)NC(C)CCCNC(=O)C=C2CCC2)cc1[N+](=O)[O-] C(=O)(C1CCc2cccc(=O)n21)N(C)CC1CCCN(C(C2(OC)CC2)=O)C1 N1(C(Cc2cccc(OCC)n2)=O)CCC(C)N(C(=O)C(C)CC(F)(F)F)CC1 c1(OC)ncc(C(=O)Nc2cccc(C#N)c2)cc1C1=COCC1 C1(C)(NC(C(N2CC(OC)C(C(=O)NCC(F)F)C2)=O)=O)CCC(=O)N(C)C1 CCCCCC(O)CC(=O)N(CCCC(=O)NCC(O)COC)C C1(C)(C(=O)NC2CCC(NC(CCC(C)(C)C#N)=O)C2)COc2ccccc2O1 N1(C(c2ccn(CCC)n2)=O)CCC(C(=O)Nc2csc(C)c2)CC1 Cc1cc2sc(C(=O)NC3CC4CC(NC(=O)CCCF)C3C4)cc2s1 c1(OC)ccc(C(O)C(N2CCC(CCNC(C3C4COCC34)=O)CC2)=O)cc1 Cc1ccc(F)c(S(=O)(=O)C(=O)O)c1.c12ccc(cc1[N+](=O)[O-])CS2 C(=O)(CS(C)(=O)=O)NCC1C(NC(CCCOC(CCC)=O)=O)COC1 N1(C(N(C2(c3ccccc3)CCOC2)C)=O)CCN(CC(C)(C)O)C(C)(C)C1 c1(C(N(C(CCNC(CC(=C=C)C)=O)C)C)=O)cccc2nc(CO)[nH]c12 c1(N(CCCNC(C(=C)Cl)c2cccs2)C)ccc(C)cc1 C1(O)(C(=O)NCC2(C(=O)NC)CCC(NCC)CC2)CC(C)CC(C)C1 C1(NC(CCNC(C)=O)=O)CCCCC12CN(c1nccn3nnnc13)CCO2 C1(C(N(C2CCCCC2)CC)=O)CC2(C)CCC1(C)O2.c12cccc(c1)NC2=O CC1(NC(c2cc(-c3ccccc3)ns2)=O)CCN(C(=O)Cc2cncnc2)C1 CC1(C)CN(C(c2ncccc2O)=O)CC1NC(c1ccnc(CO)c1)=O C(CCC(=O)NCC1CC1)NC(C1CCN1C(C1(c2ccccc2)CC1(F)F)=O)=O N1(C(CCC)=O)CC2(CCCN(C(=O)CC=Cc3ccc(Br)cc3)C2)C1 CC1(C)CCCCC(C(=O)NC2CCCC(NC(c3cocn3)=O)C2)C1 CCCCCCC(C)CC(=O)NCc1cn(CCOCC2CCCCC2)nn1 C1(CNC(C(C)(N(C)C(c2csc(CO)n2)=O)C2CC2)=O)CC(O)C(O)C1 C1(CNC(=O)CCNC(c2ccco2)=O)CCCCN1C(=O)CN1CC2CC2C1 C#CC1CN(C(c2cc(C)sc2C)=O)CCN(C(=O)C(=Cc2cccnc2)F)C1 c1(C(=O)NCC(=O)NCC2CC2NC(=O)C(C2CC2)C2CC2)cccc(F)c1 Cc1nc(C(=O)NC23CC(C2)N(C(=O)Cc2ccc(F)c(F)c2)C3)ccc1C#N c1(OC)cnc(NC(c2ccc(C3CCN(CC(F)F)CC3)cn2)=O)nc1 Cc1c[nH]c(C#N)nc1=NCCCCCNC(C1(F)CCS(=O)(=O)C1)=O N1(C(=O)C=CC2CC2)CCC2CN(C(C3(F)CC3c3ccccc3)=O)CC12 c1(C(=O)NC2CC3CC(C2)N(c2cc4ncnn4cn2)C3)ccc2nn[nH]c2c1 S(=O)(=O)(c1cccc(C(=O)NC2CN(C(=O)CC3CCC3)CC2C)c1)NCC#C C(CC(CO)NC(c1cc(CNC(c2coc(C(C)C)n2)=O)on1)=O)OC Cc1ccc2c(c1Br)CCCN2S(=O)(=O)c1cccnc1NCc1n[nH]c(C)n1 C1(NC(C=Cc2cn(C)nn2)=O)COCCN(C(c2ccnn(C)c2=O)=O)C1 c1(C(N(C2CCN(C(CCC=CC(C)C)=O)C2)C)=O)cnc2ccnn2c1 CCCCC(CC)C(=O)NCC1CC(O)CN1C(=O)Cc1ccc(C2CC2)cc1 C1(C(=O)NCC2(F)CC(CNC(Cc3c(C)n(C)cn3)=O)C2)CC(C2CC2)=NO1 CCCCC(C)C(=O)N(CC(C)NC(c1cnc(C2CC2)o1)=O)C Cc1ccnc(O)c1C(N1CC(O)(CCNC(c2ncsc2C(F)(F)F)=O)C1)=O Cc1n[nH]c(C)c1CCC(=O)NCC1C(C)CCN1C(c1cnccn1)=O CC(C)(C(=O)NC1CCCCC1Nc1nc(Cl)ncc1Cl)C(F)(F)F C(=O)(CCCS(N)(=O)=O)NC1C(NC(C(C(C)C)n2ccc(C)c2)=O)CC1 C1(OC)CN(C(c2c(C)ncn2O)=O)CC1NC(c1cc(Br)n(C)n1)=O n1(CC#C)cccc1C(=O)NC1(c2ccccc2)CC(NC(C2CC2Cl)=O)C1 N1(C(C2(CC=C)CCOC2)=O)CC2(CC(C(=O)Nc3ncccc3CC)CO2)C1 C1(NC(c2cc(C)sc2)=O)CCCC(NC(=O)CC2CC(n3cnnc3)C2)CC1 N1(C(=O)NCc2c(C)nns2)CCC2CCNCC2C1 C#Cc1ccc(C(=O)NC(CN(C)C(c2oc(Br)cc2C)=O)CC)c(C)c1 C1(NC(c2cc(C)ncc2)=O)CC2CC(NC(C3(F)CCCCCC3)=O)C2C1 C=CCC(C)(C)CC(=O)N1CC2CC1CN(C(c1cnc(C(F)F)nc1)=O)C2 c1(C(C(=O)NCCNC(=O)OC(C)(C)C)N(CCC=C)C)nscc1Br c1(-c2cn(C3(C(C(C)CCCCO)=O)CC3)nn2)cc(F)c(F)cc1F C1(C(N2CC(C(=O)OCC)C2)=O)(NC(=O)CCc2ncnn2C)CC(CO)C1 c1(C(N2CCC(CN3N(c4nnc(CC)o4)CCC3)CC2)=O)cc2ccsc2[nH]1 C1(NC(C2CC(C)OCC2)=O)CCN(C(=O)Cc2ccc(O)cc2Cl)C1(C)C C1(O)(CCNC(C2C(C)CC2)=O)CN(C(=O)Cc2csc(C(C)(C)C)n2)C1 CCC(CC)(CO)C(=O)N1CC2CCC(CNC(C3CCCC(OC)C3)=O)C2C1 C1(C(N(CCO)CC)=O)CCN(C(=O)CC2COCC(C)O2)O1 N1(C(c2c(C)cccn2)=O)CCOCC12CCN(C(c1cnc(Br)s1)=O)C2 N1(C(c2noc(C)c2C)=O)CCC12CN(Cc1ccc(C(F)(F)F)nc1Cl)C2 CC(C)(C(=O)NCCC1CS(=O)(=O)C1)C1=CCNC1 C1(CC(=O)OC)CC(OC)CN(C(=O)OC)C1.c12ccc(o1)c(=O)[nH]2 C1(C(C)NC(c2nc(CC)sc2)=O)CCCN(C(=O)Cc2cnccc2C)C1 O=C1NC2(CNC(C3C=CCN3C(=O)Cc3ccc(O)cn3)=O)CCC1C2 C1(CCOC)(NC(c2ocnc2C)=O)CCN(C(=O)C(C)OCC(C)C)CC1 CCC(CC)C(F)C(=O)N1CC(O)(CCNC(=O)CCSc2ccccc2)C1 C1(C)(NC(CCOCCCOC)=O)CCN(C(C2(O)CC2(C)C)=O)CC1 CC1CN(C(c2c[nH]c(=O)cn2)=O)CCC1C(N1CCC(N=[N+]=[N-])C1)=O c1(C(=O)NC23CC(NC(c4cnc(-c5ccccc5)[nH]4)=O)(C2)C3)ccc(=O)oc1 N1(C(C2C3CC2N(Cc2ccc(Br)c(F)c2O)C3)=O)CCn2cccc2C1 O(NC(=O)C(CNC(=O)C(C)N(C)C)OC)CC#C CN1CCC(CCNC(c2coc(CNC(=O)CC3CCCCO3)c2)=O)C1=O c1(C(=O)NC2CN(C(c3ccc(F)cn3)=O)CC2(F)F)ccc(F)c(Br)c1F c1(N(CCN(C)C(c2ccc(CO)cc2F)=O)C)[nH]c(=O)n(C)c(=O)c1C#N Cn1c(=O)cc(C(N2CCC2CNc2ncccn2)=O)c2ccccc12 Cc1cc(C(N2CCC(C)(CNC(=O)CN3CCCNC3=O)C2)=O)[nH]c1C C#Cc1ccc(C(=O)NC(CNC(c2n[nH]cc2F)=O)C2CC2)cc1Cl Cc1cnc(C(=O)NC2CCCCC2CC(N2CC(F)C(F)C2)=O)c(F)c1 c1(C(=O)NC(C(=O)NCC(CSC)OC)(C)CO)cc(C)nnc1C c1(C(=O)NCC2(C)CC2C(=O)OC)cncc(C(C)(F)F)c1.C1(CO)CCCN1OC C#Cc1c[nH]nc1C(=O)NCC1C2CN(C(c3ccc(CN(C)C)o3)=O)CC12 Cc1cc(C(N2CC(F)(CNC(=O)C(C)C=Cc3ccccc3)C2)=O)nn1C CC(=O)C(C)CC(C)C(=O)N(C)CC1CCCCN1C(C1CNC(=O)O1)=O C(=O)(CCCCCCS(N)(=O)=O)N1CC(NC(C(C)CC(F)(F)F)=O)C(O)C1 c1(C2C(n3cc(CN(C(c4oc(CC)c(C)c4)=O)C)nn3)C2)ccc(Cl)c(F)c1 C12(C(=O)NCCCCCNC(=O)Cc3ccccc3F)CSCC1C2(F)F C1(C(=O)OC)CCC(C2CCCCC2)CN1c1nc(O)c2ccccc2n1 C1(C(=O)NC2CC(CC)CC2O)(CNC(C2(CO)CCCO2)=O)CC(F)(F)C1 C1(C(=O)NCCSCCO)(CC)CN(C(=O)Nc2ccncc2)C1 N1(C(CCN(CC)CC)=O)CCC2(CCCN2C(=O)CCC2=CCCCC2)CC1 N1(C(CC2N(C(c3c(OC)cccc3)=O)CC(F)C2)=O)CC(C)N(CC)C(C)C1 C1(NC(C2CN(C(C)=O)C2)=O)CC2CCC(C1)N2C(=O)CCCCN(C)C C(C)(C(C)COC)(c1nnnn1CCN1CCCOC1)NCc1scc(CC)n1 N1(C(c2c(OC)csc2)=O)CCCC(CNC(c2ccc(C(C)=O)cn2)=O)C1 N1(C(C2(CC=C)CC2)=O)CCC2CCCC(C1)N2c1ncnc2sc(CC)cc12 N1(C(=O)C(F)CC2CCOC2)CC(C(=O)NCC2(O)CCC2)C(O)C1 C1(c2n(C(C)C3CC3)nc(-c3ccncc3)n2)CN2CCN1CC2 N#Cc1cc(CSCc2cc(Cl)cc(Br)c2)cc(Cl)c1 N1(C(C(CCC)NC(C2C=CCS2)=O)=O)CCC2(CCCN2C)C1 O=C(CCCCNC(C1CCCCC1)=O)NCC1(CCO)CCCC1 c1(CN(C2CCOC2)C)ccc(F)cc1Br C(=O)(C(F)(F)C(F)F)NCC(C1CC1)NC(c1ccc(CC(C)C)cc1)=O CC1CC(C(=O)N(CC(=O)N(C)C)C)N(C(C23CSCC2C3)=O)C1 C1(CNC(C2N(C(C=C(CCC)CCC)=O)CCC2)=O)CCC(C)(C)CO1 CC1OCCC1CN(C)C(C1(C)CN(C(C2CCC2(F)F)=O)C1)=O c1(C(=O)NCC2C(CNC(c3ccc(CC)nc3)=O)C2)sc2ccsc2c1C CC1OC2(CO)CC1(NCc1cc(C(=O)O)n[nH]1)C2 c1(C(=O)NCC2N(C(c3ncn(C)c3)=O)CCC2(C)C)cnc2nccnc2c1 c1(C(N2C(C)(C(=O)Nc3cc(C)nn3C(C)(C)C)CC2)=O)cc(F)c(Cl)nc1Cl C1(N(C(CC(C=C)C)=O)C)CN(C(c2cc(C)cc(C)c2)=O)CC12CC2 Cc1nc(=NC(=O)C2(F)CCN(C(c3ccc(-n4cncn4)nc3)=O)C2)s[nH]1 C1(CNC(C2(SC)CCC2)=O)CCN(C(C2CSCN2C)=O)C12CC2 N1(C(c2cncc(CC)c2)=O)CCC2(CCN(C(=O)CN3CC(F)(F)C3)CC2)C1 CC(Cc1ccccc1)C(C(=O)Nn1ccnn1)N1CCCCC1COC(F)F C1(CNC(=O)CC(F)F)CN(C(c2cc[nH]c2)=O)C2CC12 c1(C(N(C2CCN(C(C3C=CCC3)=O)C2)CCO)=O)cccc(F)c1F Cc1nnc(C(C)NC(c2conc2CNC(c2ccnn2C)=O)=O)s1 C1(CNC(c2ccn(CCCC)n2)=O)CC(NC(=O)CCCOC)C1(C)C C1(C(NOCCCC#C)=O)CCc2ccccc2NC1=O CCC(C(=O)OC)C(=O)N1CCCN(C(=O)NC2C3CCC23)CC1 c1(C(N(C2CCN(C(C3CC3F)=O)C2)CC)=O)nc2ccccc2[nH]1 C1(NC(c2cncc(CC)c2)=O)CC(O)CN(C(=O)Cc2cccc(C)c2)C1 C1(C2CN(C(C(C)OC)=O)C2)CN(C(=O)CCCCF)CCO1 C(=O)(CCCCC(N)=O)N1C(C)(C(=O)NCCc2n(C)cnn2)CCC1 CC1CCC(OC(F)C(=O)N2CC(NC(=O)COC(F)F)C2)CC1 c1(NC(c2c(Br)c(C)n(C)n2)=O)cc(-c2nn[nH]n2)cc2[nH]ncc12 C1(CNC(CC(C)(F)F)=O)C(C2CC2)CCN1C(c1nnc(Cl)cc1N)=O C1(CNC(c2ccn(CC)n2)=O)CN(C(c2ccc(=N)[nH]n2)=O)CC(C)(C)O1 C(=O)(C(C)(C)CC1CCC1)N(N(CCCN1CCOC1=O)C)C c1(OC)c(C(=O)NC2CCC(CCNC(=O)CN(C)CCO)C2)c(C)nn1C c1(C(=O)NCC(CNC(c2ccc(O)nc2)=O)OC)cncc(-n2cnnn2)c1 C1(C(=O)NC2CN(C(C34CC5CC3C4C5)=O)CC2C)(COC)CC=CCC1 C(=O)(C(Cn1ccnn1)NC(=O)CCOC1COC1)NCCC1CC(CC)C1 C1(CC)(NC(=O)CN(C)C(C)C)CCCN(C(c2ccnn2C(F)F)=O)C1 C1(C(N)=O)CCC(C(=O)N(C2CCCN(C(=O)C(F)F)C2)CCO)CC1 Cc1cccc(OC(C)C(=O)NCCOCCNC(c2c(C)[nH][nH]c2=N)=O)c1 C1(C)(CNC(c2c(C)cn(C)c2)=O)CN(C(C2CCN2S(C)(=O)=O)=O)CCO1 CC(C(C)(C)C(=O)NCC1(C)C=CCCC1)NC(=O)C(O)C1CC1 C1(C(=O)NC2(CC=C)CCN(C(=O)C(C)SC(C)C)C2)(OC)CCCC(C)(C)C1 CC(C)C(C(=O)N(C(C)C(C)(C)C)C)C(C)NC(C1CN2CCC1C2)=O Cc1ccc(C(=O)N(C)C(c2cccnc2)C)c(C2CC2)c1 C1(CC)CCN(C(=O)CN=[N+]=[N-])C1CNC(=O)C(C)OCCOCCO c1(OC)nccc(C(=O)NCC(C)=CC(=O)N(CC(N2CCCC2)C)C)n1 c1(C(=O)NCCC(C)NC(C2N(CC)C(=O)CC2)=O)ncn2ccccc12 Cc1cccc(C=CC(N2CC3CC3(CNC(C3CCC(C)(C)C3)=O)C2)=O)c1 c1(C(N2CC3CCN(C)CC3C2)=O)cc2c(F)c(F)c(F)cc2[nH]1 C(=O)(CC(C)Cc1ccc(Cl)cc1)NCC(C)N(C(COCCC)=O)C c1(SCC)cnccc1C(N1CCC(CO)(CNC(=O)C(C)CC)C1)=O n1(CC(N2CCC(N)(Cc3ccccc3)C2)=O)ccc2nc(O)nc(O)c12 N1(C(C(C)C#N)=O)CCC(NC(c2c(Cl)cccc2Br)=O)C(C)(C)C1 C=CC(CCC)CC(=O)NCC1CN(C(c2nn(CC)cc2Cl)=O)CCN1C c1(C(N(CCN(C(SS(C)(=O)=O)=O)CC)CC)=O)cc[nH]c(=N)n1 CC1CC(C(=O)NCC=C2CCN(C(C3CCCC4CC34)=O)CC2)=NO1 c1(SC)ccc(CCC(=O)NC2CC(C)(NC(=O)COC3CCCOC3)C2)cc1 C1(NC(COCCCCC)=O)CS(=O)(=O)C2CN(C(=O)C(C)(C)CF)CC12 c1(-c2ccnc(OC)c2CO)ccc2c(c1NCc1ccc(Cl)o1)OCO2 c1(NC(CC(C)NC(C23CC(C2)C3)=O)C)nccnc1C#N C1(NC(c2cccc(C)n2)=O)CC2CCC(C1C)N2C(C1CCCCC1(F)F)=O C(CC1=CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1)NC(Cn1ccc(C)n1)=O Cc1cccc2c(C(N3CC(NC(=O)CSc4nncs4)CC(O)C3)=O)c[nH]c12 c1(C(C(=O)NCC2N(C(COC)=O)CCOC2)N(C)C)cc(F)cc(F)c1 N1(C(C(C)C2CCCC2)C(=O)NCC2CCCO2)CCC(C2CCOC2)CC1 c1(C(N(C2CN(C(c3c(C)coc3)=O)CC2(C)C)C)=O)cc(F)c(F)cc1F c1(C(N2CCCC(CN(C(=O)CC3(C)CCCO3)C)C2)=O)csc2nccn12 Cc1nc(O)nc(C)c1CC(=O)N(C)CCNC(c1cc(Br)cnc1N)=O N1(C(CC2(CC)CCC2)=O)CCC(CNC(C2C=C(C)CS2)=O)C1(C)C c1(OC)cccc2c1OCC(C(=O)NCC(F)CNC(=O)CS(=O)(=O)N(C)C)C2 CCC(CCC(=O)N1CCN(C(=O)C(=Cc2cccc(Cl)c2)C)CC1CC)SC C1(CNC(CSc2onc(CC)n2)=O)CCN(c2nnc(C3CC3)o2)CC1C c1(C(=O)NC(C)CN(C(=O)CC2CCCCC2(C)C)C)cc2cncn2c(O)n1 c1(C(N2C(CNC(c3nc(C)c(C)s3)=O)CCC2)=O)cnn2ccn(C)c12 N1(C(=O)COC2CCC2)CCC(C(=O)NCC2CCOCC2)(CF)C1 c1(C(=O)NCC2CCCC(NC(C(=O)NCC)=O)C2)cnc(OC)cc1C(F)F N1(C(CCC(C)(F)F)=O)CCCN(C(=O)CCc2cncc(O)c2)CCC1 C(=O)(C#CC1CCOCC1)N1CCCC(NC(CC(C)C(C)(C)C)=O)C1 CC#CC1CCN(C(=O)C(CNC(C2(Cl)CCC2)=O)OC)C1 C12(C(N(CCCF)CC)=O)CC1CN(C(=O)C(C1CCC1)OCC)C2 N1(C(CSCC)=O)CCN(c2cn(C(C)CO)nn2)C(=O)C1 c1(C(=O)NCC2(NC(C3(N(C)C)CCCC3)=O)CCCCC2)cc(O)cc(Cl)c1 c1(OC)cc(Br)cc(NC(C23CC2CN(C(=O)C(c2ccc(Cl)cc2)C)C3)=O)n1 C#Cc1cccc(CC(=O)NC2CC(F)(CNC(C3CC3NS(C)(=O)=O)=O)C2)c1 c1(CNC(c2cc(OC(F)F)ccc2[N+](=O)[O-])=O)ccccc1S(=O)(=O)C(F)F CC1(CNc2ccc(N3CCNCC3)nc2)CCCCC1(F)F C1(CN(C(c2nc(CC)sc2)=O)C)CN(C(=O)C(O)CC)CC12CC2 N1(C(CC2N(CC)C(=O)CC2)=O)CCCC(C2CCN(C(=O)CC(F)F)CC2)C1 c1(C(N(CC(C)NC(=O)Cc2ccc(F)cc2F)C)=O)ccc(F)c(CO)c1 N1(C(C2CC23CC(O)C3)=O)CC2(CO)CC1(C(=O)NOCCCCC1CC1)C2 Cc1ccsc1C=CC(=O)NCCCNC(C1CC12CC2(F)F)=O Cc1nnc2n1CC(C(=O)NCCC1(NC(=O)C(O)C3CC3)CCC1)CC2 CCC(CC(=O)NC1CCCCC1NC(=O)C(c1nc(C)cs1)C)OC C1(NC(c2c(C)c(C3CC3)on2)=O)CC2CC1CN(C(=O)C(C)C(F)(F)F)C2 CC(C)CC(C)C(=O)NCC1CC(F)CN1C(c1coc(C2CCCCC2)n1)=O C1(C)(COC)CC(NC(c2nc(CO)cs2)=O)CN1C(=O)CN(C(=O)C(C)C)C C1(C2C(=O)N2CC(C)C)CCC1(C)C.CCC(C)(C)NC(=O)OC(C)(C)C C(=O)(CC(CC)CC(C)C)NCC(CCC)NC(=O)COc1ccsn1 c1(C(N(C(C)Cc2ccc(F)cc2F)C2CC2)=O)c(Cl)cccc1Br c1(C(=O)NCC(C)(C)NC(C2C(C)(CC)C2)=O)ccccc1OCCN(C)C C(=O)(C(O)CC(F)(F)F)N.C(C(COC)CC(=O)N1CC(SCOC)C1)OC n1(CC)nnnc1C(C(C1CC1)OC(C)C)NCc1nc(C(C)(C)C)cs1 C(=O)(CCCN=[N+]=[N-])N(CCN(C(=O)CCc1ccccc1C#N)C(C)C)C c1(C(N)=O)ccc(SCC(=O)NC2CCCC2NC(c2cnc(Cl)[nH]2)=O)cc1 c1(C(N2CCN(C(c3ccc(CCC)[nH]3)=O)CC2)=O)ccc2c(c1)C(C)CN2 C1(C(=O)OC)CCCC(NC(=O)C(c2ccc(Cl)cc2)N(c2ccnc(Cl)n2)C)C1 N1(C(COC(CC)C)=O)CCCCCC(NC(c2cnc(Cl)c(N)c2)=O)C1 CN1C(=O)NCC12CN(C(C1CCCN(C(c3ccc(F)nc3)=O)C1)=O)C2 C(=O)(C(C(=O)N(C(C)CNC(c1cccc(=O)o1)=O)CC)C(C)(C)C)OCC C1(C(=O)NCCCOCCC(=O)NC(C(C)C)(C)C)C2CCCOC12 N1(C(=O)Cn2cc(C3CCC3)nn2)CCC2(CCCN2C(C2COC2)=O)C1 c1(OCC)ccc(C(=O)NC2CC(C(=O)NCC3CCOCC3)C2)cc1Cl C1(C(N(C)Cc2nc(C)on2)=O)CC12CCN(C(c1scnc1Cl)=O)C2 C1(NC(c2snc(Cl)c2Cl)=O)CCCN(C(=O)C2=CCCC2)C1 C(=O)(C(C)(C)CC(F)F)NCC1C(NC(CCNC(=O)NC)=O)C1 N1(CC(=O)NCC)CCC(CC2CN(C(c3[nH]nnc3C)=O)CCO2)CC1 N1(CC(CO)NC(=O)Cc2ccsc2Br)CCCCC1 C1(O)(CNC(c2cccnc2OC(F)F)=O)CCN(C(c2ccco2)=O)C1 Cc1c(C(=O)NC(C)CC(C)NC(c2nncn2C2CC2)=O)ccn1C c1(C(=O)NCCC2CC(NC(C(C)SCC)=O)C2)cc(C(N)=O)[nH]n1 CC(CC(=O)NCC1CC1CC(=O)Nc1cn[nH]c1)n1cccc1 C1(C(N2C(C3(O)CN(C(c4cc(Cl)ns4)=O)C3)CCC2)=O)CCc2nnnn2C1 C(CN=c1[nH]c(=NCC2CCc3ccccc32)[nH]c2cccc(F)c12)OC(=N)O C(c1cccc(F)c1)=C(C(N1C(CNC(c2c(C)csc2Cl)=O)C(C)CC1)=O)F C1(NC(c2cc(OC)ncc2)=O)CCCN(c2nccc(OC)n2)C1C c1(C(N2CC(CNC(C3C(C)(CC)C3)=O)C2)=O)cc(C)nc2ccccc12 c1(OC)ccc(C(=O)NCCC(C)NC(=O)Cc2ccnn2C)cc1.C1CN1 C=CC1CN(C(C2CC(=O)OC2(C)C)=O)CC1C(=O)NCC CCCC(F)(F)C(=O)N1CCC(C)(CNC(=O)CCCC2CC2C)CC1 c1(CC(=O)NCCc2cn(C3C(SC)CCC3)nn2)ncccc1C c1(NC(C2(F)CCN(C(Cc3nc(C)on3)=O)C2)=O)cc(F)ncc1F C1(NC(CCC(=C)C)=O)CC(OC)CN(C(C2CCC2C(=O)OC)=O)C1 CS(=O)(=O)c1cccc(N2CCCN(c3ccncc3)CC2)n1 C=CCC(CC(=O)NC(c1cscn1)C)NC(C1CCC1(F)F)=O C(=O)(C(CSc1nc(-c2ccc(C(F)(F)F)cn2)no1)CC1CCCC1)OCC N1(C(c2[nH]cc(C)c2)=O)CCCC2(C1)CN(C(c1ccc(NC=O)cc1)=O)C2 C1(NC(C2(OCC)CCC2)=O)CCN(C(C2CCC(C)=C(C)C2)=O)CC1F Cc1cc(C(=O)NCC(CO)NC(c2cnc(N(C)C)o2)=O)c(C)n1C1CC1 S(=O)(=O)(c1ccc(NCC(F)F)cc1)N1CC(O)CCC(C)C1 c1(CN(C(c2ccc(I)cc2)C(=O)O)C)cc2c(Br)cccc2o1 C(=O)(CS(=O)(=O)NC(c1cccc(NC)c1)=O)OCCN(C(C)=O)CC c1(NC(C2N(C(c3cc(C(C)(C)C)ncc3)=O)CC2)=O)ncc(Cl)nc1Cl C=CC(O)(C(=O)N1CCC(C(=O)NCCC2(N(C)C)CCCC2)CC1)C(F)(F)F C1(NC(CCOCC#C)=O)CCN(C(C2(CC3C=CCCC3)CC2)=O)CC1 C1(C)(C(=O)NC2CC(N(C(C(c3cnccn3)C)=O)C)C2)CC2(CCC2)C1 Cc1c(NC(=O)CC(C)CNC(=O)OC(C)(C)C)cccc1[N+](=O)[O-] CCC(CC)C(=O)N(CC(C)(C)CNC(=O)Cc1cccc(F)c1)C C1(C(=O)NC(C2CCCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)C)CS(=O)(=O)CC(=O)N1 Cc1cc(C(=O)NC2(C(N3CC(c4nncn4C)C3)=O)CCCC2C)nn1C C1(C(=O)NCC(CSC)(F)F)CCCCCN1C(=O)C=CC1CCOC1 C1(Cc2scc(C(N3CC(NC(C(CC)OC)=O)C3)=O)n2)CCS(=O)(=O)CC1 C1(F)(CNC(=O)Cc2cccnc2)CC2CCC(C1)N2C(C1CC(C(F)F)C1)=O Cc1nocc1CC(=O)N(CCCCCNC(c1sccc1Cl)=O)C(C)C CCN(OC)C(=O)CC(C1CC1)NC(=O)CCCCCF N1(C(C(CCC)O)=O)CCCCCC1C(=O)Nc1cccc(OC)c1O Cc1cc(F)ccc1C(O)C(=O)N1CC(N(C)C(c2c(C)ncn2C)=O)C1 c1(C(=O)NCC(CC)NC(C2COC3(CO)CC2C3)=O)nn(C)c(C)c1Br C1(C(=O)NC(CCCNC(C(C(=C)C)(C)C)=O)(C)C)CC12CCC(C)(C)CC2 N1(C(COC(C)C)=O)CC2CCCCC2(CNC(C2CCCC2F)=O)C1 c1(C(=O)NCCN(C(C=CC(C)C)=O)CCOC)cnn(C(F)F)c1 c1(OC)cc(C(=O)NC2(CC(=O)NCC3CC34CC4(F)F)CCCCC2)ccn1 C1(NC(CCc2ncc(C)[nH]2)=O)COC2(CCN(C(C3CCCC3O)=O)CC2)C1 C1(CNC(=O)CC(C2CC2)C2CC2)CCCN(C(c2cc(Cl)ncc2F)=O)CC1 c1(C(=O)NCC(N(C)C(c2cncn(C)c2=O)=O)C2CC2)n[nH]c2ccccc12 C1(C(=O)NC(C2CN(C(c3ccc(C)nc3)=O)C2)C)CC12CCOC(C)C2 C1(N(C(=O)CCN2CCC2)C)CCCCN(C(c2ccc(Br)c(N)c2)=O)C1 C(C(F)(C(=O)NC(c1nc(C)oc1C)C)C(C)C)NC(CC(C=C)(C)C)=O N1(C(C2CC(C#C)(O)C2)=O)CCCC(C(=O)NOC(C)CC)CC1 N1(C(C2(C#C)CCN(C(=O)C=CCF)CC2)=O)CCOCC(C2CC2)C1 C(=O)(C(C)CCCOC)NC(CCC)C(=O)N1CC(C)(C(F)(F)F)C1 C1(CC(=O)N)CCC2(CCC2)O1.C=CCCC(=O)NC(CCC)C1CC1 C1(NC(C(CSC)n2cccn2)=O)COCCC1NC(C1CC(C(C)C)C1)=O N1(C(CC(C)CN(C)C)=O)CCC(O)C(N(C(=O)C(C)(C)C2CCCC2)C)C1 C(=O)(C(C)(C)CNC(c1cccnn1)=O)NC(c1cscn1)C CCC(CC(C)C)C(=O)N1CCC(NC(c2cnc(OC)cn2)=O)C1(C)C c1(C(N(CCCOCCNC(C2(CC)CCC2)=O)C)=O)nn2ccccc2c1C C(=O)(CCCC(F)(F)F)NC1CCCN(C(C(CC)C(=O)OCC)=O)CC1 c1(N(C(C(C)=C(CC)C)=O)C(=O)CCSc2ccc(C)cc2)ccc2c(c1)OCO2 C1(C(N2C(C)CCC(CNC(c3cnc(S)nc3)=O)C2)=O)CC2(CCCC2)CO1 N1(C(C(=O)Nc2nccc(CCC(=O)OC)c2)=O)CC2CC(C1)C2O C12(CC=C)CCCN1C2=O.c1(C(C(=O)N(c2cccnc2)CC)O)cccnc1 c1(C(N2CCC(OCC(=O)NC(c3cnnn3C)C)C2)=O)ncccc1F Cc1nc(C)n(CC(N2C(C(=O)NCC(C)(C)C(C)C)CCC2C2CC2)=O)n1 c1(C(=O)NCC(N(C(CN(CCC)C)=O)C)C2CC2)cc([N+](=O)[O-])nn1C N12CCCC3(CCN(C3)NC1=O)C2.C1(CC(CN(C)C)=O)CCCS1(=O)=O c1(C(N2CCCC(N(C(=O)Cc3ccon3)C)C2)=O)nc(O)nc(O)c1N Cc1noc(C)c1C(=O)NC1CCCC1CNC(c1nnn(C2CCOC2)c1C)=O C=CCC(C)C(=O)N1CCCCC1CC(=O)N(C1CSC1)C C1(C(=O)N(C(C2CN(C(=O)CCc3cncs3)C2)C)C2CC2)CCCCC1C1CC1 C12(C(N3C(C(=O)Nc4n(C)nnc4)CC4CC43)=O)CC3CC(CC(C3)C1)C2 N1(C(C(C)CN(C)C)=O)CC(CNC(c2cnn(C)c2N)=O)OC(C)(C)C1 N1(C(C2N(C(CC3C(C(=O)OC)C3)=O)C(C)C2)=O)CCCCC(CO)C1 C(=O)(C1=CCCC1)NC1(C(=O)NC2CCC(SC)C2)CCCC1 C(CNC(=O)C(F)CC1CC1)(C(C)(C)C)NC(C(c1ccccc1)N(C)C)=O C1(C(=O)NCC(=C)C)CN(C(C2C3CCC(C3)C2C)=O)C2(CCC2)C1 C1(CCNC(c2ccc(CCC)[nH]2)=O)CCCN(C(C2(CC)CC2(F)F)=O)CC1 CCC(C)(C)CC(=O)N(C(C)C(=O)Nc1cccc(OC)c1)CC C(N=c1[nH]nco1)c1n(Cc2cn(C3CC3)nn2)ccn1 Cc1ccnc(-c2nnc(C(C)OC(CCC(C(C)C)c3ccccc3)=O)o2)n1 Cc1nc(Cl)cc(=NC(C)C2CN(C(C3(O)CCSC3)=O)CCO2)[nH]1 Cn1nc(C(=O)NC2CN(C(C3(O)CCC3)=O)CC2C(F)F)c2c1CCCC2 c1(OC(C)C(=O)NCCC(C)N(C(=O)CC(=O)OC2CC2)C)cccnc1 Cc1cc(C(=O)NC2(C)CC(C(=O)NCCNC3CCCC3)C2)cs1 c1(C(=O)NC2CCN(C(c3ccc(C)c(Cl)c3)=O)C(C)C2)ccc(F)c(F)c1F C(=O)(C(C)(C)CCC(C(=O)NC1CCCC1)N(C(C#N)C1CC1)CC)OCC C(C(O)CC(C)(O)C(F)F)OCCNC(C)CF C(c1cnc[nH]1)=CC(N1CC(O)(C2CCCN2C(C2CCCO2)=O)C1)=O N1(C(=O)Cc2cccnc2F)CCC2(CC1)CC(N1CCCCC(O)(CF)C1)C2 CCCCC(C(=O)NCc1cc(C(=O)NCCC(F)=C(F)F)no1)N(C)C C1(C(=O)NC(C)CNC(=O)CC2CCOCC2(C)C)CC12CCc1ccccc12 C1CC2=CCN(C2)C(=O)C(C)O1.C(CNCC1CC1)=CC Cc1c(NCC2(CO)CC(F)(F)C2)ncnc1NC1CCCOC1C(C)C N1(C(c2ccn(C)c(=O)c2)=O)CCC2(CCCN2C(=O)CCc2cncs2)C1 N1(C(C(CSC)OC)=O)CCC(C(C)C(=O)NC(C(C)(C)NC(C)=O)C)CC1 C1(CC(=O)NC2(COC)CCN(C(CN(C)CCO)=O)C2)COC(C)(C)CO1 N1(C(=O)NCCC2CCCCO2)CCC2CC2C1 CNS(=O)(=O)N1CCC(C(=O)NCC2COCCN2C(=O)CCF)CC1 N1(C(C(CCC)CNC(=O)C(C)CC(C)CC)=O)CCC2CC1C(=O)N2C C=CC(CC)CC(=O)N1CCC(OCCC2CCN(C(c3cnco3)=O)CC2)C1 c1(C(=O)NCC2(O)CCCN(C(C3C(C)OCCC3)=O)C2)ccc2nsnc2c1 C(=O)(C1=NOC(C)C1)NC1(CNC(C2C(CC)C2)=O)CCOC1 C1(C)(C(N2CC(COC)(CNC(=O)COC3CC=CC3)C2)=O)CC=CCO1 c1(CNC(C2C(C)C2C)=O)ccccc1C#N.C12CCN(CC1)C(=O)CNC2=O CCCCCC(C)(C)C(=O)NC(C)CCCNC(c1coc(-c2cccs2)n1)=O c1(NC(C(c2cnc(C(C)C)s2)N(C2C(SC)COC2)C)=O)ccc(C)c(C)c1 c12ccc3[nH]cc(c3c1)CN2.c1(C)cccnc1C(=O)O.O(CN(C)CC)O C(CCC(N)=O)(C(=O)N(C1CN(C(c2c(C)cccc2Cl)=O)CC12CC2)C)OC n1(CC)ncc(C(=O)NCC2(F)CN(C(c3nccnc3C)=O)C2)c1Cl c1(C(=O)NCC(CCCC)NC(=O)CSCC=C(C)C)cncc2c[nH]nc12 Cc1ccc(C)n1CC(N1CCC(NC(c2ccc(F)s2)=O)C1C)=O Cc1nn(CCC(=O)NC2CCCC(NC(C3(O)CC3)=O)C2)cc1Br C(C(C)(C(C)C)NC(c1nnn(C(C)C)c1C)=O)NC(CC1(COC)CC1)=O C1(C(N(C)Cc2cncs2)=O)(CNC(=O)Cc2ccns2)CC12CCC2 C1(C(=O)NC2CC(CNC(CC=C(C)C)=O)C2)CCOCC12CCC2 c1(CN2CC3C(C(=O)Nc4cc5n(n4)CCC5)C3C2)cc(Cl)cc(Br)c1O C1(NC(CCCNC(C)=O)=O)CCN(C(c2cnns2)=O)CC1(C)C N1(C(C2C(C)CCO2)=O)CC2(CCN(C(=O)C(C)(C)NS(C)(=O)=O)CC2)C1 Cc1ccc(SCCC(=O)NC2COCCC2NC(C2(C)CCC(=O)C2)=O)cc1 c1(-n2c(C(C)SC)nc(-c3ccncc3)n2)ccnc2c1cnn2C C#Cc1ccc(C(=O)N(C)CCN(C(=O)C(C)OC2CCCCCC2)C)c(F)c1 C1(F)(C(N(CCOC)CCNC(=O)CCc2nccn2C)=O)CCC(C)CC1 N1(C(C(C)=CC)=O)CC2(C)CN(C(c3cnn(CCOC)c3C)=O)CC2(C)C1 N1(C(C(C)CC(N)=O)=O)CCC2(CC(NC(C3(CCCF)CC3)=O)CO2)C1 c1(NC(c2ccccc2)C(=O)N(C2CCCN(C(C)C)C2)C)ccc(Cl)cc1 C1(C(=O)NC2(C#N)CCC2)CCN(S(=O)(=O)Cc2ccc(F)cc2)CC1 c1(CC(N2CC3(C(NC(COCCC)=O)CC3)C2)=O)ccc2nc(O)[nH]c2c1 FC1(F)CC(n2nnnc2C(CC2CCOCC2)NC2CCOC2C2CC2)C1 c1(OC)cc(Cl)cc2[nH]c(C(=O)N(C)CCOCCSc3cncs3)cc12 C(=O)(CC(C)C(C)C(C)C)NCC1OCCCN(C(CCc2onc(C)n2)=O)C1 C(=O)(CC(C)(C)CC(F)(F)F)NC1CCCCN(C(C2(C(=O)NC)CCC2)=O)C1 C(C(O)CC(=O)N1CCC1(C)CC(=O)NC1CN(CC(F)F)C1)N(C)C CC(Cc1ccccc1)C(=O)N(C)CCOCCNC(C1CC1(C)Br)=O C1(NC(c2nc(CC(C)C)sc2)=O)CCC2CN(c3nnc(C(F)F)s3)CC2C1 C1(C(=O)NO)CCCC(C(F)(F)C(F)F)N1.C1(C)CNC1 C1(O)(CCNC(C(C)CO)=O)CCCN(C(c2n[nH]c3c2COC3)=O)C1 S(=O)(=O)(c1cccc(F)c1)N1CCCC2(N(C(c3cnc[nH]3)=O)CC2)C1 C1(CC=C)(NC(C2CCCSS2)=O)CCN(C(=O)CCc2cc(Cl)cs2)CC1 C(CCCCC(=O)N1CCC(OCCCNC(C2CCC(F)C2)=O)CC1)=CC c1(C(N2CC(CCNC(C3C(C(C)(C)C)C3)=O)C2)=O)cncc(CO)c1 C(=O)(C(C)CCCOC)N(C(CN(C(COCc1ncc(C)o1)=O)C)C)C CCCCCC(F)C(=O)NCCCCC(C)NC(c1cnc(CC)nc1)=O C1(OC)(CNC(=O)Cn2ncnn2)CN(C(C2(Cl)CC2(F)F)=O)C1 C1(C2CCN(C)CC2)(C(=O)NCC2N(C(C(C)OC)=O)CC(OC)C2)CC1 C1(CC)CN(Cc2cnc(O)c(Cl)c2)CC2(CCOC2)O1 N1(C(CC2C(C)CCC2)=O)C2CCC1CC(CNC(c1cccc(F)c1)=O)C2 N1(C(C(=O)N(C(C)C)CCO)C)CCN(C(=O)COC2(C)CCOCC2)CC1 N1(C(CC)=O)CCN(C(=O)CCOc2ccccc2Cl)C(C)C1C N1(C(C(=O)N(C)C)=O)CC2(CCN(C(C3(C)C(C)(C)C3(C)C)=O)CC2)C1 N1(C(c2c(C)noc2C)=O)CCC(C)(NC(C2(c3ccc(O)cc3)CC2)=O)CC1 c1(C(N(C)CCN(C)C(C2CC3CCC2C32CC2)=O)=O)ccc2ncccc2c1 N1CCOCC(C(=O)NCC2CN(S(=O)(=O)C(F)F)C2)C1.CCCC(=O)OC c1(CN(C(c2ccccc2)C(=O)NC(C)CC)CC)cccnc1.C1C(=O)N1 N1(C(C2=NOC(CNC(Cc3c(C#C)cccc3)=O)C2)=O)CCC(O)CC(C)C1 c1(C(=O)NCC2CC(NC(C(C)N(C(C)=O)C)=O)C2)cc(Cl)ccc1F C1(CNC(CC(C=C)(C)C)=O)CCC2(CCC2)C1NC(c1cccc(Cl)c1)=O Cc1cc(C(N2CC3(C2)CN(C(=O)C(O)CC2CCOCC2)C3)=O)cc(O)c1 Cc1nc2ccc(C(=O)NC3CN(C(=O)CSS(C)(=O)=O)CC3F)cc2[nH]1 CCN=C(NCC(c1ccccc1Br)OCC1CCC1)NC1CSC1 C1(NC(=O)Cc2cc(C3CC3)no2)CCCCC1NC(c1cc(C2CC2)no1)=O Cc1ccncc1CC(=O)NC(C)CC(C)NC(=O)C=CCN(C)C1CC1 C1(C(=O)NC2CCC(CCNC(CCc3cc(OC)no3)=O)C2)CN(C)CCO1 c1(C(N2CC(C(N3CCC(N(C)C)C3)=O)C2)=O)cc(Cl)c(Cl)cc1Cl c1(C(=O)NC2CCN(C(C3CC3(F)Cl)=O)C2)cc(=O)cc[nH]1 C1(NC(CC2CCC(C)O2)=O)CCC(N(C)C(c2ccn(C3CC3)n2)=O)CC1 c1(CC)ccc(C(=O)NC2CCCC2NC(=O)C(O)C2CCC2)c(OC)c1 N1(C(=O)CNc2onc3c2CCCC3)CCC2(CCCNC2)CC1 CC1CCN(C(c2cnc3n2CCS3)=O)C(CNC(C2(O)CC3CCC2C3)=O)C1 C1(C(=O)NC(CC)CN(C)C)CC(O)CCN1C(C1C=CCS1)=O C(=O)(C(O)P(C)(C)=O)NCC(C)NC(c1c(C2CCC2)cnn1C)=O c1(CNC2C=C(C)CCC2)cc(C)c(Cl)c([N+](=O)[O-])c1 O=C(C1=CCSC1)N1CC2CC1(C(=O)Nc1cncc(F)c1)C2 c1(CCCC)cc(F)c(S(=O)(=O)N2CCCC(NC(C)=O)C2)c(F)c1 c1(COC)ccccc1NC(=O)CN1CCC(C)CC1.N12CC(C)(C1)OCC2 c1(NC2CSCN(C(=O)OCC)C2)cc(N=[N+]=[N-])ccn1 C1(C(N(C(CCNC(Cc2cc(C(=O)OCC)sc2)=O)C)C)=O)CC=CCC1C c1(C(=O)NC2CC(NC(c3ccnc(OC)n3)=O)C2)ccc2cnoc2c1 C1(CNC(c2cn(CC)nn2)=O)(CNC(c2c(CC)non2)=O)CCCCC1 C1(C(C)C)CN(C(c2ccnc(C3CCC3)c2)=O)CCN1C(=O)OC(C)(C)C Cc1cc([N+](=O)[O-])cnc1C(N1CCN(C(=O)Cc2ccoc2)CC1C(C)C)=O C(CC(C)C)(C(=O)NCCC(=O)NO)NC(CC(COC)C)=O C1(CNC(C(CC)C)=O)CC2(CC2)CN1C(=O)COc1cccc(C#N)c1 C1(C(=O)NCC2(F)CC(NC(C(CC=C)NC(C)=O)=O)C2)CCCC(F)(F)C1 c1(C(N(C)CCNC(c2ccc(N3CCCC3)cc2)=O)=O)ccc2c(c1)CCCO2 c1(C(N(CCCCO)C(C)C)=O)ccc(CNC(C2COC(C)C2)=O)o1 CCCCCCCNC(=S)Nc1ccccc1N1CCN(CCC)CC1 C1(CC)C(C(=O)NCC(Cl)C(C)(F)F)CCN1C(=O)CSC(C)C c1(C(N2CCOC(C3CCC3)C2)C)ccc(Cl)cc1 c1(N(C)C)cnc(CNCC(C)(C)NC(C2(C3CCCCO3)CCC2)=O)cn1 c1(N(CC(=C)Br)C)nc(N2Cc3c[nH]nc3C(C)C2)nc2c1CSC2 CC1(C)CC(O)(C(=O)NCC2CCCC(CNC(c3cnc(C#N)s3)=O)C2)C1 C1(C(=O)NCC(c2ccccc2)N(C)C(c2ccccn2)=O)OCCN(C)C1=O C(O)(C(F)(F)F)C1(C(=O)NCCCN(C(=O)CCc2nncs2)C2CC2)CCC1 CN1C2CCC1CC(CC(N1CCC(F)(CNC(C3CC3F)=O)CC1)=O)C2 C1(=CC(=O)NC(C(C)NC(Cc2c(C)n[nH]c2C)=O)C)CCOc2ccccc21 O=C1CCc2ccc(CN3CCC4(CC4C(=O)N=c4ccc(Cl)n[nH]4)C3)nc2N1 c1(C(N2CCCC(C#C)(O)C2)C(=O)NCC(C)C)noc2c1CCCCC2 C(=O)(CCCCCCN=[N+]=[N-])N(C1CC(NC(c2ccc3cnoc3c2)=O)C1)C CC(C)C(F)C(=O)NC(C(=O)NC1(C)CC2(CC2)C1)C1(C)CC1 C(CCOCCO)(C(=O)NCc1cccc(CO)c1)NC(C(CC)C)=O c1(C(=O)NC2C(CNC(CNC(N)=O)=O)CCCC2)ccnc2ncccc12 C1(CC(=O)NC2C(C(=O)NCC(C)C)OCC2)CCC(C)(C)C1 C(C(C(=O)NCCC(C)O)C(C)C)NC(c1c(C)nc(C)o1)=O CC#CCC(C(=O)NC1CCCCC1(F)F)NC(c1cc(C)nc(O)c1)=O C1(C(N(C)CCNC(c2cncc(N3CCCC3)n2)=O)=O)CCC(C)(C)OC1 Cc1c(N)ccc(C(N2CC(NC(c3ncc(F)cn3)=O)C3(CCC3)C2)=O)c1Cl C1(NC(c2ccc(F)s2)=O)CCCN(c2nnc(-c3ccon3)s2)C12CCCC2 Cc1cc(Cl)c(Cl)cc1C(N1CCC(O)(CN(C(=O)COCC2CC2)C)CC1)=O C1(NC(=O)NCCCN(S(C)(=O)=O)C)CCC(=O)N(CC2CC2Cl)CC1 N1(N(C(c2noc3ccccc23)C=O)C)CCC(C2(O)CC2)CC1.C1(C)CCC1 CCCCCCC(C)C(=O)N1CCN(C2CN(C(C3(C)CCC(=O)C3)=O)C2)CC1 c1(NC23C(CN(C(=O)OC(C)(C)C)C2)CC3)cnc2cccnn12 C(=O)(C(C)(C)C(O)C(C)C)NCC(CC)NC(c1cc(O)ncn1)=O C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)(C(C)C)NC(C)=O C1(N(C(=O)CC2CCSC2)CCNC(C(C)(C)OC)=O)CCCCCC1 CC1(CNC(=O)CNC=O)CN(C(c2sccc2Br)=O)CCO1 c1(C(=O)OC)cc(C(=O)N(CC(O)CNC(c2ccc(SC)cc2)=O)C)c(C)o1 CC(CCN=c1nc(N(CCC(=O)N(C)C)C)c2[nH]ccc2[nH]1)N(C)C C1(O)(CNC(CN(C(C)C)C(c2cc(CCO)on2)=O)=O)CCCOC1 C1(CC(=O)NCCC2CN(C(=O)C(CO)N3CCCCC3)C2)CN2CCC1CC2 C1(CC)CN(C(=O)CC2(COC)CC2)CCC1NC(=O)Cn1cnc(Br)c1 c1(CNC(C2C(C)(CC)C2)=O)cn(CCNC(c2cscn2)=O)nn1 N1(C(=O)CCOC(F)(F)F)CCCCCC1C(N1CCOC(CF)C1)=O C1(NC(CCCC=C)=O)COC2(CCN(C(C3(c4cccs4)CC3)=O)C2)C1 c1(C(=O)NC(CNC(C(n2ncc(C)c2)C)=O)C(C)C)sccc1S(N)(=O)=O N1(C(Cc2cc(C)sc2)=O)CCC(CF)(NC(C2CCOC(C(C)C)C2)=O)C1 Cc1nc(C)c(C(=O)NC2CN(C(C3(c4ccc(O)cc4)CCOCC3)=O)C2)o1 Cc1nc(C(N2CCOCC2CC(C)C)C(=O)NCC2CCCO2)oc1C C1(C(N2CCCC(CCC(=O)NC3(C)CCSC3)C2)=O)(CC)CCCCO1 C=CC1(C(=O)N)CCN(C(=O)CCCC(=C)C)C1.C(CC(=O)N)CCSC(F)F CC1(C)CCC2(CC1)CN(C(=O)C(F)C(F)(F)F)C2 CC1(C)NC(=O)N(CC(N2CC(NC(=O)C3=NOCC3)C(F)C2)=O)C1=O c1(C(N(C(CNC(CC(CCC)(C)C)=O)C)C)=O)cnn2ccc(Cl)c(F)c12 C1(NC(C2CCC(C)O2)=O)CCN(C(c2ncc(F)cn2)=O)C(C)C1 C1(NC(C2C(=C)C2)=O)CN(C(c2ccccc2-n2cccc2)=O)CC1(C)C c1(C(N(CCCNC(=O)CCCCC2CC2)CC)=O)ccc2cc(C)ccc2c1 C(=O)(CC(F)(F)CC(=O)NC1CC(NC(c2ccc(C)nn2)=O)C12CCC2)OC C(=O)(C1Cc2ccc(F)cc21)NCCC(CNC(C=Cc1cnc(C)s1)=O)O C1(NC(=O)COC2CCN(C(=O)CC3CCCCCC3)C2)CCCCCC1CO c1(OC)cc(C(N2CCC(NC(c3cc(=O)c(OC)c[nH]3)=O)C2)=O)cc(Cl)c1 c1(C(CNC(c2ccnc(C)c2)=O)NC(CC(C)OC)=O)ccc(F)cc1F C1(CNC(c2cc(C)ns2)=O)CCN(C(=O)C(C)Cc2ccccc2C)C12CC2 c1(C(=O)NC(C2CCCN(C(=O)OC)C2)C)ccc2c(c1)CCOC2 C1(C(N(CC(=O)NCC(C)Cc2cn[nH]c2)CC)=O)CCC(F)CC1 n1(CC)ncc(C(=O)NC2CCCCC2C(N(C)C[Si](C)(C)C)=O)c1C C(C1=CCCN(C(=O)CC2CC(O)C2(C)C)C1)NC(c1c(C)n(C(C)C)nn1)=O C1(NC(c2cc(C)ns2)=O)C=CCC(C(=O)Nc2cccnc2)C1 N1(C(C2N(C)C(=O)CC2)=O)CCC2(CC1)C(NC(C1CCOC1)=O)CS2(=O)=O c1(SC)nc2ncnc(N3CCC(CNC(C4(C)CCCCNC4=O)=O)C3)c2s1 C(CC(=O)NCCOC1CN(CCO)C1)N(C)CC.S(S(C)(=O)=O)CC(=O)N Cc1[nH]nc(C(N2CCOC(C(=O)NCc3ccco3)C2)=O)c1O N1(C(C2(OC(C)=O)CC2)=O)CCN(C(c2cc(O)n(C)n2)=O)C(C2CC2)C1 N1(C(COCCCC)=O)CCC(C2CN(C(c3csc(CO)n3)=O)C2)CC1 C1(C)(CNC(Cn2nnc(C)n2)=O)CN(C(c2c(O)noc2C)=O)CCO1 C=Cc1cc(C(N2CCC3(NC(=O)CCCOCC)CC3C2)=O)cc(F)c1 C(N=c1nc(Oc2cccc(C)c2C)cc(C)[nH]1)c1ccc(OCCC)c(F)c1 C(=O)(C1CCCc2sccc21)NCC1CN(C(C2C3(CC(C)(C)C3)C2)=O)C1 c1(C(=O)NC(C2(O)CN(C(=O)C=CC3CCOC3)C2)C)ccc(F)c(Cl)c1F N1(C(C(c2cn(C)nc2)=O)=O)CCC(NC(=O)C=C2CCN(C)C2)CC(O)C1 c1(CNC(C2CC(NC(Cc3cn(CC)nc3)=O)C2)=O)c(Cl)cccc1Cl C1(C(C(=O)NC(CC=C)CO)F)CCC(F)(F)CC1 CCC(CC(=O)N1CC(OC)C1)OCCC(=O)N(C)CC1(F)CCCC1 N1(C(C2(CC)CCC2)=O)CC2CC(C)N(C(c3cc(C)c(C)cc3C)=O)C2C1 c1(C2(NC(=O)Cc3ccon3)CC2)ccc(F)cn1.C12CC(F)(C1)CNC2=O CC1CC(NC(N)=O)CN(C(=O)CCOC(=O)CC2COCC(C)O2)C1 c1(-c2nc(C(C)C)nn2C2CCC(C)C2)cc(F)cc(F)c1Br CC(C)(C)CC(O)C(=O)NC1CC(CNC(C2(Oc3ccncc3)CC2)=O)C1 S(=O)(=O)(c1cc([N+](=O)[O-])cc(Cl)c1F)Nc1c(C(=O)OC)ccnc1 S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C)N1CC(CNC(c2c(C)ncc(C)n2)=O)C1 Cc1cc(C(=O)NCC2CN(C(=O)CC3C=CS(=O)(=O)C3)CC2O)nn1C1CC1 c1(CNC(=NCC)NCC(c2ccc(F)cc2)O)nc(Br)c(C)cc1Cl C1(C(=O)NC(c2ccc(C)cc2)CC)CC(NC(=O)CN2CCOCC2)C1(C)C c1(N2CC(C)(C3CC3)OCC2)ccc(Br)c(S(=O)(=O)N2CCCC2CF)n1 C(=O)(C(C)(C)C(=O)N1CCC(C(C)(C)CNC(C2CC2(F)Cl)=O)CC1)OC c1(NCC2(NC(CNC=O)=O)CC2)ncnc2[nH]cc(C)c12 C=CC(CCC)CC(=O)NC(CC(C)(C)C)C(=O)NC1CCC(C)(C)C1 C(F)(F)(C(F)C(F)(F)F)Oc1cccc(C(=O)OC(C)CCC(F)(F)F)c1 N1(C(c2ccc(CCCCC)o2)=O)CCC(C)N(c2cc(O)nc(O)n2)CC1 C#CC1(NC(c2cc(CNC(C3CCOC3C=C)=O)no2)=O)CCC(C)(C)C1 c1(C(=O)NC2C(NC(C(CC)N(CC)CC)=O)C2)cc(NC(N)=O)ccc1Cl N1(CCO)CCC2CN(c3c(C)noc3COC(C)(C)C)CCC12 CCCC(C(F)(F)F)NC(C1CC(O)CN1C(=O)COc1ccc(C)cc1)=O C1(C(=O)NCCC=CC=C)CCN(C(=O)C=C(C)COCCOC)CC1(C)C CC1(C)COC(C(=O)NCCC2CCN(C(=O)Cn3cc(Cl)cn3)C2)CO1 C(CCC(=O)N(C(C)CN(C(=O)Cn1nnnc1C)C)C)=C(C)C CC(C)(O)CCN=C(NCc1sccc1Br)NC1CCCC1 c1(OC)cc(C(N2CCCC2C(=O)Nc2ncccc2[N+](=O)[O-])=O)cc(F)c1F c1(C(N2CCSC3CCCC23)C(=O)NC2(C)CC2)ccc2c(c1)CCC2 C1(NC(C2CCN(Cc3cnn(CC)c3C)C2)=O)CN2CCC1CC2 Cc1cc(NC(C2CCCN2C(=O)CN(C)C(N)=O)=O)cc(Br)c1C N1(C(C2C(OC)CN(S(=O)(=O)C3CC3)CC2)=O)CCCC(C2CCCNC2)C1 C1(NC(=O)CNC(c2cccs2)=O)CC2CCC(C1)N2C(=O)CCn1cccc1 c1(N(CCOC)CCOC(=O)Cc2cncnc2O)ccc(OC)c(C)c1 C(c1ccc(F)c(Cl)c1)=CC(N1CCC(C)(NC(c2cc(C)cc(Cl)c2)=O)C1)=O c1(C(N(CC(C)O)CCNC(C2CC(O)(CC#C)C2)=O)=O)cnccc1C CC1CN(C(=O)CCC(F)F)CC(C)N(C(c2cc(Cl)c(Br)cn2)=O)C1 c1(NC(C(Cn2cncn2)NC(=O)Cc2ccsc2)=O)ccc2n[nH]cc2c1 Cc1cc(CCC(=O)N(C2(CC(=O)NCCCOC3CCC3)CC2)C)on1 C1(NC(CC2C=NN(C)C2=O)=O)CN(C(=O)CN(C2CCSC2)C)CC1C1CC1 CCCC(CC)CCC(=O)NCC(C)CNC(=O)CCc1nccn1C C1(=CC(=O)N(C(CC)C(=O)N(CC)Cc2cnc[nH]2)C)CCC(C)CC1 C1(C(=O)NC2C(NC(CC3CCC(C)(C)CC3)=O)C2)CC2CSCC(C1)C2 Cc1[nH]c(C)c(C(N2CCCC(CCNC(=O)COc3ccsn3)CC2)=O)c1C C1(C)(C(N2CC(C(N(CCN(C)C)CCO)=O)OCC2)=O)CCCCC1(F)F C1(C(=O)NCC2CC(NC(C(C)OC)=O)C2)CCCN2CCCCC12 C12(NC(=O)COCC3CCC3C(=O)NC3CCCO3)CC3CC(CC1C3)C2 c1(C(N2CCCCCC2C2CC2)C(=O)NCC=C)nc(Br)ccc1F C(=O)(CCC(CF)CF)N1CCC(C(C)C(=O)NCCCNC(=O)C2CC2)CC1 Cc1cc(Cl)c(C(N2C3CC2CN(C(=O)COCc2nc[nH]n2)C3)=O)cc1C C1(NC(=O)C=CCF)COCCC1NC(c1csnc1Cc1ccccc1)=O CCCC(C#N)C(=O)N1CCC(NC(c2ccc(C)nc2OC)=O)C(CC)C1 CC1CN(C(C2(CSC3CC3)CCC2)=O)CCN1C(=O)COc1ccc(F)nc1 C1(OC(COCC)=O)CN(C(=O)CC2(COC)CC2)CCC1C Cc1c(F)ccc(C(N2CC(C)(C)CC2CNC(=O)CCCNC(N)=O)=O)c1N C1(CNC(c2ccc(C)cc2)=O)CCN(C(=O)C(C)OC2CCCC2)C12CC2 CCCCC(O)CNC(=O)C(C)CN(C)C(c1nocc1C(C)C)=O C(=O)(C(F)CC(C)(C)NC(=O)CN1CCCCC1=O)OCC.C1(N)CCC(CC)CC1 c1(C(N2C3CN(C(C(CC(C)(C)C)O)=O)C(C3)C2)=O)coc2c1C(=O)NCCC2 c1(CCC)cnnc(C(=O)NCC(O)CNC(C2CC=CCC2)=O)c1 c1(CC)ccc(CC(=O)NC(CNC(c2nn(C)cc2C)=O)C2CC2)cc1 c1(SC)cc(C(N2CCCC2CNC(C2CC3C(C2)C3(F)F)=O)=O)ccc1F C(=O)(CC(C)(C)C(F)F)N(C(CC(=O)N(C(c1ccco1)C)C)(C)C)C c1(OC)cc(O)ccc1C(=O)NC1CC(C(=O)NC(C)CN(C)C)C1 c1(C(=O)NC2CN(C(C(C(C)C)=O)=O)CC(C)C2)ccnc2cc[nH]c12 c1(C(=O)NC(CC=C)C(=O)NCCN2CCCCCC2)ncnc(O)c1F C(c1cccc2ccccc12)=CC(=O)NCC(C)(O)C(F)(F)F C1(C(=O)NCC2C(NC(CCCC=C)=O)C2)CCc2c(cnn2C)C1 C1(C(=O)OC)Oc2ccc(NC(=O)NC3CC4CCC(C3)C4(C)C)cc2C1C N1(C(C(C2CC2)OCC)=O)CCN(C(c2cc(C(=O)OC)[nH]n2)=O)CC1 c1(-c2nc(C(N3CCC(O)(COC)C3)=O)sc2)csc([N+](=O)[O-])c1 c1(OC)nc(C(=O)NCC2CCC(F)(CN)CC2)ncc1F c1(CC)cc(Cl)ncc1CNC(c1ccccc1F)c1ccccc1 c1(C(N2C(C)CCC(NC(=O)C=C3CCCC3)C2)=O)c(F)cc(N)cc1F N1(C(C2CCC(C)O2)=O)CC(NC(C2CCC(c3ccccc3)O2)=O)C(C)(C)C1 c1(C(N2CCCCC(N(C(C(CSC)C)=O)C)C2)=O)occ2c1CCOC2 C(CC(=O)NC1CC(C(C)NC(c2csnn2)=O)C1)SCCCC CON=CC(=O)NCC1CC(NC(=O)C(C)c2ccsc2)C1 C1(CNC(CCC)=O)CCN(C(=O)Cc2nn(C)cc2Cl)C(C)C1 N1(C(c2cc(CC)ncn2)=O)CC2CC(NC(=O)C(F)(F)c3csc(=N)[nH]3)C1C2 N1(C(C2(CC)CC2)=O)CCC(C2CCCN(C(C3CCC=CO3)=O)C2)C1 c1(C(N2CCC(N(C(=O)CC3CCC(C(F)(F)F)O3)CCO)C2)=O)cccc(Cl)c1 C1(NC(CSC)=O)CC(CNC(=O)C(N2CCNC2=O)C)C1(C)C C(=O)(C(CC1CCCO1)C(F)(F)F)N1CCC(CCNC(C=NOC)=O)CC1 c1(C(N2C(C)CC(NC(=O)Cc3cn(C)cn3)CC2)=O)nc2ccccn2c1F N1(c2nc(C(=O)OC)c(C)s2)C(CNC(C2CC2F)=O)CC2COCC12 c1(C(=O)NCC2(CO)CC3(CC(F)C3)C2)cnn2ccc(F)cc12 C1(C)(NC(C(C)N(C(=O)CN2CCCCC2)C2CC2)=O)CN2CCC1CC2 C1(NC(c2ocnc2C2CC2)=O)CCCCCC1C(=O)NCC(F)Br C1(CC(=O)NC2CC(NC(c3ccc(C)o3)=O)CC2O)CCCCC1(C)C N1(C(C(C)NS(C)(=O)=O)=O)CCCC(C2CN(C(c3cnc(S)nc3)=O)C2)C1 c1(OC)ccc(C=CC(=O)NCC(C)(O)CNC(C2(C)CC(F)C2)=O)cc1 N1(C(C(CN(C)C)O)=O)CCC(C(C)(C)NC(=O)C=Cc2cncn2C)CC1 c12ccc(c(OC)c1)OC2.C(=O)(C(=O)NCC1CC(CC(F)F)C1)NCC c1(NC(C2CCC(NC(COCC(=C)C)=O)CC2)=O)cccc(CC)c1O C12(C(=O)NCC(CC)NC(C3(C)CCCS3(=O)=O)=O)CCC(CO)(CC1)C2 C1(CNC(C2C(OCC)C2)=O)CN(C(=O)CCNc2ncccn2)C2(CCC2)C1 c1(CN(CC)CC)ccc(C(=O)NC(C)CCNC(=O)Cc2ccno2)o1 c1(C(=O)NCC2(CNC(Cn3c(C)ccn3)=O)CCCC2)sc(=N)[nH]c1C CCCC(CNC(c1ccc(Br)cc1)C1CC1)CCC CC1CN(C(=O)COc2ccc(C(F)(F)F)cc2)CCC1NC(C1CC(F)(F)C1)=O N1(C(C2CN(CC(C)C)C2)=O)CC2(CCN(C(C3CC4CCC3C4)=O)CC2)C1 C#CCCCC(C)C(=O)NC12CC(NC(c3cc(O)cc(F)c3)=O)(C1)C2 c1(OC)ccc(OC)c(C(=O)CCC(=O)OCCCCC2(C)OCCO2)c1 C(=O)(CCCC1CCC1)N1C(OCC(=O)NCC(CC)n2cccn2)CC1 C#CCC(CC(=O)NCCCc1nnnn1C)NC(C1CCCC1O)=O c1(CN(C2CC(C(=O)NC(c3ccco3)COC)C2)CC)ccccc1 C1(N(C(=O)CCn2ccnc2)C)CCN(C(=O)COc2cccnc2)C1 c1(C(N2CCC(C(C)NC(=O)CC(F)(F)F)C2)=O)cc2ccsc2s1 c1(OC)cc(C)ccc1CNCc1ncc(SCc2ccccc2)nc1C C(=O)(C1CCc2nnc(C)n21)NCC(C)(C)NC(c1cc(C)[nH]c1C)=O C12(CNC(CC=CCNC(CC#N)=O)=O)CCCN1CCC2 N1(C(C(C)SCC)=O)CC2CCC(C1)N2C(c1sccc1-n1cnnn1)=O c1(C(N2CCC(O)(C(C)NC(CCC)=O)C2)=O)cc([N+](=O)[O-])cnc1N CCCCCCCCC(F)C(=O)NCC1CN(C(C2CCC(C)O2)=O)CC1(C)C C1(C(=O)NC2CC3CC(OC)C3C2)COC2(C1)CN(C(c1cscc1Cl)=O)C2 C=CCC(C)(CC)C(=O)NCC1C(CNC(c2c(C)coc2C)=O)C1(F)F C(=O)(C(F)(F)F)NCC(=O)NCCC1CN(C(=O)CC2CC(F)C2)C1 C1(N(C(=O)CC(=O)OC(C)(C)C)CC)CCN(C(c2cnsn2)=O)CC1 C(C)(CO)(C(=O)N1CCCC(CNC(c2cnc(N(C)C)s2)=O)C1)NC(=O)OC C12(SC)CCC(CC1n1cc(CC3CC(c4ccon4)C3)nn1)C2 C1(CC)C(C(=O)NCCSC)CCCN1C(=O)C#CC1CC1.C(=O)C(C)OC c1(C(=O)NCC2CCN(C(C3(C)CCOCC3)=O)CC2)cc2ccccc2cn1 C(=O)(CCCCC(=O)N1CC2CCC2(CNC(=O)CCC2CCOC2)C1)OC C1(NC(C2C(C3C(C)C3)C2)=O)CC2CN(C(=O)CCCn3cncn3)CC2C1 n12cc(nn1)C2CC.c1(C(=O)NC(CSC)CC)ccccc1 C1(NC(N2CC3C(C(N4CC(N(C)CCO)C4)=O)(C3)C2)=O)CC2C=CC1CC2 c1(C(C)OC(CC)CNC(=O)C(=O)Nc2ccccc2)cc(Br)ccc1Cl C(=O)(C(O)P(C)(C)=O)NC(C(C)(C)C)CNC(=O)C=CC(F)(F)F CCC(C)(C)CC(=O)NC(C(=O)NCC1(C)CCN(C)C1)C1CCCO1 c1(CCC(=O)NC2C(NC(C=C(C)C)=O)CCC2)c(C)nc(S)nc1C c1(C(=O)NC2CN(C(CCc3ccc(OC)cc3)=O)C2)cc(=NC2CC2)cc[nH]1 N1(C(C(C(CC)CC)OC)=O)CC2CCCC(C1)N2C(=O)C(C)C#N CC(C)(CNC(C1(Cl)CC1)=O)CC(=O)N1CCC(CN=[N+]=[N-])C1 c1(C(=O)NC(CC)CNC(=O)C#CC2(CC)CC2)ncc(C#N)cc1C C1(CNC(c2c[nH]nc2-c2cccc(Cl)c2)=O)CCCCN1C(c1ccon1)=O c1(OC)ccnc(C(=O)NCC2CCCN(C(c3ccc(C(F)F)s3)=O)C2)c1O N(C1CCCn2ccnc21)C(C(C1CC=CCC1)NC(c1ccnc(O)c1)=O)=O Cc1cc(-c2ocnc2C(=O)NC2CC(NC(=O)CC3CC4CC4C3)C2)on1 N#Cc1ccc2c(c1)CN(C(=O)CCc1cc3ccccc3[nH]1)C2 CC1CCN(C(=O)CC2CC3(CC3)C2)C1C(=O)NCCn1ncccc1=O c1(CCNC2(C(=O)OC)CCN(C(=O)NCC(=O)OC)C2)ccc(OC)cc1 C(=O)(C(CC1CC1)OC)NC1CC(C(N2CC(C(=O)OCC)C2)=O)C1 C(CN=c1nc(C)cc(C)[nH]1)n1cc(-c2cncc(C(=O)OC)c2)nn1 c1(C(N(C2CCCN(C(C=CC)=O)C2)C)=O)ccc(-n2cccn2)c(F)c1 CC1CN(C(=O)C2=C(Cl)CCC2)CCN(C(C2(C)C(C)(C)C2(C)C)=O)C1 N1(C(Cc2cc(OC)no2)=O)CCC(C)C(NC(=O)CCN2CCC(F)C2)C1 N1(C(C(C)NC(=O)OC)=O)CCC(O)(CNC(=O)CC2CCCC(C)(C)O2)CC1 CCCC(C(=O)N1CCC(N(C(c2cc(Cl)ns2)=O)CC)CC1)N(C)C Cc1cnc(NC2(CO)CCCCC2)c(S(=O)(=O)NC2CC3CC(O)C2C3)c1 C(=O)(CC(C(=C)C)OCC)NCC(CC=C)NC(=O)Cn1nccc1C CS(=O)c1ccccc1C(=O)NCCC(O)CNC(=O)CCc1ccccc1 CC1(NC(C2CC(=O)N2)=O)CCN(c2ccnc(C#N)n2)CC1 C12(NC(c3c(C)sc(O)n3)=O)CCCC(NC(C3CCCC3C)=O)(C1)C2 C(=O)(C1Cc2ccc(Cl)cc21)N1CC(C(C)C)N(C(=O)Cc2ccccc2)CC1 C(N=c1[nH]c(C(F)F)n[nH]1)c1nnn(C(C)(C)C)n1 N1(C(CCC(=C)C)=O)CCC2(CC1)CN(C(=O)C1=CCCSC1)CC2CO C(CO)(C(=O)NC1CC(CN(C)C)C1)NC(C1C(OC(C)=O)C1)=O.C(CF)S CC1(C)CCN(C(=O)CC(C2CC2)NC(C2CCOC2)=O)CCO1 C(=O)(CC(C(F)F)NC(C1(C(=O)NC)CCC1)=O)NC(CC(=O)OC)C1CC1 Cc1cc(F)cc(C)c1C(=O)NCc1ncoc1CNC(c1cnc(Cl)n1C)=O C#Cc1cccc(C(=O)NCC(C)CNC(c2nnn(C)n2)=O)c1 Cc1oc(CNC(c2cc(C(N)=O)co2)=O)nc1C(=O)NCC1CC1C c1(NC)cc(C=CC(=O)NC2CCCCC2C)ccc1OC(C)(C)C CC(CCC(=O)NCC(C)N(C)C(c1cnc2cnn(C)c2c1)=O)S(C)(=O)=O n1(CC(=O)N(CCNC(CC(C)CF)=O)C)c(=O)oc2cc([N+](=O)[O-])ccc12 c1(C(N2CCC(CCO)C2)C(=O)NC(C)C)cc2c(Cl)nccc2s1 N1(Cc2ccn(CC(C)C)n2)CCCCC1c1ncnn1-c1ccccc1 CN=c1[nH]cc(-c2cccc3nc(C(=O)Nc4cc(C)nn4C)cn23)cc1C#N Cc1cc(C)c(C(N2CCC(CO)(NC(c3cccc(C)c3F)=O)CC2)=O)cn1 c1(C(=O)NC(C2CCOC2)CNC(c2cccnn2)=O)ccc(Br)c(Cl)c1 C1(C2CCN(C(=O)CC3CC=CCN3C)C2)(NC(C(C(C)C)N(C)C)=O)CC1 c1(CC(=O)NC(C2N(C(c3c(OC)ccs3)=O)CCCC2)C)c(C)nn(C)c1C Cc1csc2ncnc(NC3CC4CN(C(c5occc5C5CC5)=O)CC34)c12 N1(C(C2=CCC(NC(C3(OCC)CC3)=O)C2)=O)CC(O)CC(C)(C)C1 C(=O)(CC1NC(=O)c2ccccc21)N1CC(C2(NC(C(C=C=C)C)=O)CC2)C1 N1(c2cc(C#C)cc(CC)n2)CCC(C)(C)N(CC)C(=O)C1 c1(CNC(c2cnc(SC)n2C)=O)cc(O)nc(CNC(C2CCOC2C)=O)n1 c1(C(N(CCNC(C(C)(CO)NC(C)=O)=O)C2CC2)=O)cc(F)ccc1C CCCCC(C(=O)Nc1csc(C)c1)NC(=O)CCCOCCC C1(c2nnnn2C2CC2)(NC(c2ccc(C)c(Cl)c2)C(=O)OC)CCC=CCC1 CC1CCN(C(c2cc(CO)n(C)n2)=O)CC1(C)C(=O)NCC1CCCO1 C1(C(N2CCC3(C2)C(=O)N3)=O)CCC(C)=C(C)C1.C1(C(C)(F)F)(OC)CC1 c1(C(=O)NCC2N(C(c3cnc(C(C)(C)CF)o3)=O)CCC2)cccc(=O)n1O C(=O)(C1CCc2cc(F)ccc21)N1C2(CNC(CCOCCOC)=O)CC(C1)C2 N1(C(=O)OC)CCCC(C(N2CCCC2CNC(C2CC(=O)N2)=O)=O)C1 N1(C(CC(C(F)F)NC(c2ccc(C)c(C)n2)=O)=O)CC2CC1C(F)(F)C2 C(=O)(C(F)(F)C(F)F)N1C2(C(N(C)CC)=O)CC(C1)C2 NC1CCC(S(=O)(=O)NC2(c3cccs3)CCCCC2)CC1 C(=O)(C(C(C)C)Nc1cn(C(C)C)cc1C)N(CCCNC(C)=O)C Cc1csc(C)c1C(N1CCOC(CCNC(=O)C(C2CC2)C2CC2)C1)=O c1(CNC(C2CCC2NC(C2CCCN(C(C)=O)C2)=O)=O)cccc(F)c1O C1(CNC(CCCCC=C)=O)CC12CCN(C(=O)C(O)P(C)(C)=O)CC2 C=CC(CCC)CC(=O)N1CCCC(CNC(=O)Cc2ccccc2)CC1 Cc1ccc(F)c(C(N2CC3CC3C2C(N2CCC2)=O)=O)c1F CC1=NOC(C)(C(=O)NCCC(C)CCNC(=O)CCC2CCC(C)O2)C1 C1(CCC)CN(C(=O)CCCF)CC1C(=O)NCC(O)COCC c1(NC(C23CC(C(=O)Nc4nnc(-c5ccco5)o4)(C2)C3)=O)cccnc1Br C1(C(=O)NCC23CC2CN(C(C2CCCCN2C(C)C)=O)C3)(OC)CCCCC1 c1(C(N2CCCC(NC(C(CCC)CC)=O)CC2)=O)ccc2c[nH]nc2c1 C1(CS(=O)(=O)C2C(C(C(=O)C3C(CN)C3)OC)C2)CN(C)CC1(C)C c1(NCc2c(CC)nn(C)c2)[nH]c(=NCC2CC(C)(C)CO2)nc2sccc12 Cc1[nH]nc2cc(NC(C3CC3NC(=O)Cc3ccsc3)=O)ccc12 C1(OC)CCCC(NC(=O)NC2CCCC2CN(C)C(=O)OC(C)(C)C)CC1 C1(NC(C2(CC)CCN(C(c3sc(C)nc3C)=O)C2)=O)CCn2ccnc2C1 C(=O)(NNC(=O)c1csc(C(F)F)n1)NC(C)Cn1cc(-c2cnn(C)c2)nn1 C=CCC(CC(C)C)C(=O)NCCSCc1cn(CC2C3CCCC23)nn1 C1(C(N2CCC(CCNC(=O)Cc3ccc(Cl)cn3)CC2)=O)CC12CCCCC2 O=C(CCC(=O)c1ccccc1)NC1(CCCNC(c2ccc(=O)oc2)=O)CC1 C#Cc1ccc(C(N2CCC(Cc3cn(CC(O)CN(C)C)nn3)CC2)=O)nc1 c1(CN2CCC(NC(Cc3c(OC)ccc(Br)c3)=O)C2)cc(F)c(F)cc1Br c1(NC(N(C(=O)OC)CC)=O)ccccc1.c1(C2C(C(=O)CN)C2)cccs1.C1CCO1 c1(C(N2CCC(C(=O)Nc3c(C)noc3)CC2)=O)cn(C)c(=O)n1C N1(C(C(C)SCCCC)=O)CCCC(O)(CNC(=O)C2=C(Cl)CCC2)CC1 S(=O)(=O)(c1ccc(NCC(C(C)C)OCCO)c2cnccc12)NCCSC C1(NC(c2c(CCC)nsc2N)=O)CN(C(=O)CC2CC2)CC1C1CC1 C(=O)(C(C)(CC)CCC)N1CC(N2CCC(Nc3c(OCC)oc(C)n3)CC2)C1 C(=O)(CCCC(=O)N(C1CCCCC1N(C(=O)CNC(=O)C(C)(C)C)C)C)OC n1(CC)cc(C(=O)N(C)CCOCCCNC(C2(C(C)C)CC2)=O)nn1 c1(NC(C)=O)cccc(C(=O)NCC(O)CCNC(=O)C=Cc2cncn2C)c1 Cc1ccc(C(N2CC=CC(C(=O)NOCCCCC3CC3)C2)=O)cc1F CC1CC(NC(c2ccc(CC#N)cc2)=O)CN1C(=O)CN1CC(=O)NC1=O c1(COc2ccc(CNC(CC)C3CCO3)c(Cl)c2)cc(F)c(F)c(F)c1 C1(C(=O)NCCC(C)(C)CO)N(C(c2n[nH]cc2Cl)=O)CC12CCCC2 CCCCC(C(=O)NC(C)CCC(=O)N1CCCC1C(O)CO)NC(N)=O C(C)(CCC(=O)NC1CC(CCNC(c2coc(C#N)c2)=O)C1)SC c1(CNC(C2N(C(c3c(CC)nccc3)=O)CCC2OC)=O)cc(C)cnc1O C1(N(C)C)CC2(C1)CC(C(N)=O)C2.C12CC(C13CCC3)NC2 c1(OC)ccc2c(c1)C(N)CCN2C(C1CC2C(C1)C2(C)C)=O N1(C(C(CCSC)O)=O)CCCCCC(NC(C2COCOC2)=O)C1 N1(C(C)C)CCCCC1C1CCCN1.c12nccc(n1)C(=S)NCC2 c1(C(N2CCCC(C(C)NC(=O)C(C)c3ccco3)C2)=O)ccncc1N=[N+]=[N-] N1(C(C(CC2CCC2)OC)=O)CC=C(C(=O)NC(c2ccc(C)s2)C)C1 C(N=c1[nH]nc(C(F)F)s1)c1cccc(CNC(c2c(CC)oc(C)c2)=O)c1 C1(F)(CNC(C(CCC)OC)=O)CCCN(C(C2COC(=O)N2)=O)CC1 Cc1nc(C)c(CC(=O)NC2CN(C(c3cn(CC4CC4)nn3)=O)CC2C)s1 C1(C(=O)NC(c2cc[nH]c2)C)(CCNC(=O)NC2CC2)CCC1 C1(NC(CCCCC)=O)CN(C(=O)CN(C)Cc2ccccc2)C2(CCOC2)C1 C1(NC(C2(OC)CCN(C(C3CCCN3C)=O)C2)=O)CCCCCC1F Cc1ccc2c(C(=O)NC(C)CCNC(=O)CC3(N(C)C)CCCC3)csc2c1 Cc1cccc(C(=O)CSC2(C)CCCN2)c1 N1(C(C2(COCC)CCC2)=O)CC2CN(C(c3cncnc3)=O)CCC2(CO)C1 c1(C(=O)NCC(C)NC(C2(C#N)CC2n2cccn2)=O)ccc(Cl)[nH]1 c1(C(N2CC(F)(CNC(C(C)OC)=O)C2)=O)cc2ccncc2cc1F c1(C(=O)NCC(CNC(CNC(=O)NC)=O)O)cc2c(s1)CN(C)CC2 C=C(C)CN=C(NCC(c1ccc(OC)cc1)C)NC1CCCC1(F)F CC1CN(C(C2CC2F)=O)CCN1C(c1cn(CCCF)nn1)=O c1(C(=O)NCC23C(CN(C(C4C(CC)C4)=O)C2)C3)cc(F)c(F)c(N)c1Cl C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(c2cc3cscc3s2)=O)CCN1C N#Cc1cccc2[nH]cc(C(N3C(C(=O)Nc4ncccc4Cl)CC4CC34)=O)c12 Nc1ccc(C(=O)NC2CC2CNC(c2cc(=O)cc[nH]2)=O)c(Cl)c1 Cc1noc(Cl)c1CC(=O)NC1(CO)CCN(C(C2C(C)C2C)=O)C1 c1(CC)ccc(C(N2C(C(=O)Nc3ccccc3)CC3CC23)=O)cc1 N1(Cc2cn(C3CCC(C(N4CC(OC)C4)=O)C3)nn2)C(=O)COCC1=O n1(CC)nc(C(=O)N(C)C)cc1O.c12cn(nn1)C1CN(C1)C2.N12CCC1C2=O Cc1cccc2[nH]cc(CC(N3CC(C)(C)C3C(=O)O)=O)c12 c1(C(=O)NCC(C)(C)CC2CN(C(C3CC4CCC3C4)=O)C2)nc(O)nc(O)c1N C(=O)(C(CCCCC)C(C)C)NC1(CCC)CC1.C1C(=O)N1.C#CCNC(C)=O c12cc(C)nn1CC(=O)NCCNC2=O.c1(C(=O)OCC)cc(CC)on1 N=c1[nH]c(Cl)c([N+](=O)[O-])c(=NCC(O)CNC(c2cc3ccccn3n2)=O)[nH]1 C1(OC)CNCCC1CNC(C(=O)N(CCn1ccnc1)C1CC1)=O C1(C(N2CCCC2C(F)(F)F)=O)C2CC(F)C(C2)N1C(C1CCC(O)CC1)=O N1(C(c2nc(Br)ccc2F)C(=O)NCC2CCCO2)CCn2ncnc2C1 c1(C(N2CCC(CNC(C3(C)CC=CCC3)=O)C2)=O)c[nH]c2ccccc12 C(=O)(C1CNC(=O)c2ccccc21)NC1CC(NC(=O)NCCC=C)C1 C1(NC(CC(=C)C)=O)CC2CCC(C1C)N2C(=O)Cn1cc([N+](=O)[O-])ccc1=O C1(C(=O)NCC(CNC(C(c2cccc(C)c2)(C)C)=O)CO)CCC(C)(C)CC1 c1(OC)cc(N)c(F)cc1C(N1CC(N(C(=O)Cc2csnn2)C)C(C)(C)C1)=O C1(C(N(CCNC(c2nn(CC)c(C3CC3)c2)=O)C2CC2)=O)CC12CCCCC2 N1(C(C2C(C)CCO2)=O)CC(C)(C)CC1CNC(=O)Cn1cc(C2CC2)cn1 CC1COCC(CNCc2cccc(-n3ccnc3)c2)O1 N1(C(c2c(C)scc2)=O)CCN(C(c2ccc3nc(O)cn3c2)=O)C(C)CC1C CC(O)C(C(=O)N1CCC(N(C(=O)Cc2ccc(O)cc2)C)C1)N(C)C N1(C(C(C)Sn2cnnn2)=O)CC2CC(C1)CN(C(c1c[nH]nc1C(F)F)=O)C2 N(C1CCC(NC(c2nonc2N)=O)c2ccccc21)C(C(CC)(C)CC)=O c1(C(N2CCC(c3cn(-c4cccnc4)nn3)C2)=O)ccc(-n2cncn2)nc1 c1(C(=O)NCC(COC)NC(C2SCCCS2)=O)cc(OC)n[nH]1 C(C(CNC(c1ccc(O)cc1Cl)=O)C(F)(F)F)NC(C(C)(C)OC)=O CCCC(O)CC(=O)NC1CC(N(C(=O)C(c2c(C)nn(C)c2C)=O)C)C1 CCCC(C)C(=O)N1CC(NCc2nc(C(C)(C)C)no2)C(C)C1 CCC(C)(CC)C(=O)N(CC(O)CNC(=O)C(N1CCCC(C)C1)=O)C C1(C(C)(C)C2(C(=O)OC)CC2)COCCN(C(C2CC3C=CC2CC3)=O)C1 c1(C(=O)NC(CCOC)CNC(=O)CC2C=CS(=O)(=O)C2)cc(F)c(F)cc1Cl CCCC(CC(C)C(=O)NC1CC12CCN(C(C1(SC)CCC1)=O)CC2)C(C)C C1(CNC(c2c(OC)ccnc2)=O)C(C)CCCN1C(C1CC(=C2CCC2)C1)=O N1(C(CC(CC)CN(C)C)=O)CCC(N=c2[nH]c(C3CCCC3)nc(=N)[nH]2)CC1 N1(C(C2(CCNC(=O)CCCC3CC3)CC2)=O)CCCCC1CC1CC1 C1(CN(C)C(c2cccc(CO)n2)=O)CC(O)CN1C(=O)CC12CCC(CC1)C2 C(=O)(CN=c1nc2sccc2c(NC2CCOC(CCOC)C2)[nH]1)NCCCC N1(C(=O)CC2CCN(C(c3cccc[n+]3[O-])=O)CC2)CCC(F)C(F)C1 c1(C(=O)NC2CC(C)(CNC(C3(C=C)CCC3)=O)C2)sccc1S(C)(=O)=O N(C(=NCC(C1CCC1)OC)NC(C)C)Cc1ccc(CC)cc1 c1(C(=O)NC(C)CCCNC(c2c[nH]nc2C2CCOC2)=O)ccnc(S)c1 CON1CCC(NC(=O)CCN(C(=O)C2=C(Cl)CC2)CCO)C1=O C(=O)(C(C(C)(C)C)n1cc(C2CC2C(=O)OC(C)C)nn1)NCCOC Cc1ccnc(Cl)c1C(=O)Nc1cccnc1C(=O)Nc1sccc1C(=O)OC C=CC(C)(CC)C(=O)NCC1CCC(C(=O)NCc2ccnc(C)c2)O1 c1(C(N(CC(C)NC(c2c(C)nn(C(C)C)c2C)=O)C)=O)ccc2cnoc2c1 C(=O)(CC1=CCN(C(c2ocnc2C)=O)CC1)Nc1c(O)ccc(C)c1 C1(C(=O)NC(C)C(C)NC(=O)COC2CC2)(NC(C)=O)CCCCCCC1 c1(CNC(CC=CCNC(C(C)c2cc[nH]n2)=O)=O)cc(O)ns1 c1(C(=O)NC)cc(CCNC(=O)NC(C)(C)C)nn1C.C(C)(C(C(C)C)NC)C(=O)O c1(C(C(N2CC(c3cn(CC(CC)C)nn3)(C)C2)=O)(C)O)cccc(Cl)c1 C1(NC(c2c(Cl)cn(C)n2)=O)CC2CCC(C1F)N2C(c1cc(C2CC2)on1)=O C1(CNC(CNS(N)(=O)=O)=O)CCCC1NC(C1CC1C1CCCO1)=O.C1C=C1 C(=O)(CCCS(C)(=O)=O)NCCc1c(CNC(C(COC)(C)OC)=O)nco1 N1(C(C)=O)CCC(NC(C)CN(C(=O)C(=O)Nc2cccc(C)c2)C)CC1 N1(C(C(CC)C)=O)CCC(N(C)C(c2ccc(C3CC3)nc2)=O)CC1.C1CC1 CCC(O)C(C)C(=O)N(CC(O)CNC(c1cc(Br)c(C)s1)=O)C Cc1nc(CC(C)C)oc1C(N1CCC(NC(=O)C=CCOC(C)(C)C)C1C)=O C1(O)(CCNC(C2(CC)CCCCC2)=O)CCCN(C(c2ccc(O)nn2)=O)C1 C1(NC(C2(S(C)(=O)=O)CC2)=O)CC2(C1)CC(NC(C1(C)CC3CC3C1)=O)C2 C(=O)(CC(C)(C)O)NCCc1c(C(N(CCS(C)(=O)=O)C)=O)c[nH]n1 C1(C(=O)NCCCCCSC)(OC)CCN(C(=O)CSc2nc[nH]n2)C1 N1(C(CNC(CN2CCC(C)C2)=O)=O)CC(C(N2CC3(CC3)C2)=O)C2C1CCC2 c1(C(N2CC(N(C)C(C3CCC3)=O)C(C)(C)C2)=O)sc([N+](=O)[O-])cc1Cl C(=O)(CCCC(OC)OC)NCCC1(NC(CN(C)CCc2ccccc2)=O)CC1 CC1(C)CCCN(C(=O)Cc2cnsc2)C1CNC(c1ccc(O)cc1Cl)=O C1(C(N(C)CC2CCCC3CC23)=O)CCN(C(=O)CC2CCCN2C)CC1(C)C CC1=C(C(=O)N2CCOC(CS(=O)(=O)NC(=O)OC(C)(C)C)C2)CNC1 CCC(CCC(=O)N1CCCC1C1(O)CN(C(c2cc(C(C)C)no2)=O)C1)OC c1(C(=O)NC2CCN(C(c3c(C)nc(C)s3)=O)CC2O)cc2sc(C)nc2[nH]1 N1(C(C(C)SC)=O)CC2COCC(C1)C2NC(=O)CCc1cn[nH]c1 Cc1ccc2c(c1)CC(C(N1CCOC(CN(C)C(c3sncc3C)=O)C1)=O)S2 Cc1cccc(C(=O)NC(C2CCCCC2)C(=O)NCCC(C)C)n1 c1(C(N2C(C(=O)NCc3nc(=O)o[nH]3)C=CCC2)=O)ccc2c[nH]nc2c1 c1(C(=O)NCC2CC(NC(C(C(CC)C)OC)=O)C2)ccc2oc(O)nc2c1 c1(CC)cccc(C(N2CC(NC(c3sc(CC)nc3C)=O)C3(CC3)C2)=O)c1N N#Cc1ccc(CN2CC3CC3(C(=O)NCC3CCOCC3)C2)cc1 Cc1nn(C2CC2)c(C)c1CC(N1C(c2ccccc2)CCC1C1CC1CO)=O N1(C(C(CN(C)C)O)=O)CCCC(NC(C2COCC2(C)C)=O)C1 C1(CC(=O)NCC2C3CC2N(C(=O)CCOC2CC2)C3)Cn2ccnc2NC1=O C1(C(=O)NC(CNC(c2n(C=C)ncc2)=O)CCC)COc2cc(Cl)ccc2C1 c1(C(=O)NCCNC(C2N(C(CCCC)=O)CSC2)=O)cnc2c(c1)COCC2 Nc1cc(C(N2CC3CC2C3NC(c2cnsc2)=O)=O)cc(O)c1 c1(C(N2CCCC(C3CCCCN3C(=O)C=CCO)C2)=O)cnc(F)c(F)c1 c1(NC(C2CCCC2O)=O)ccc2nc(N3CCOCC3)[nH]c2c1 C1(NC(COCCOC)=O)CN(C(c2cc(OC)c(F)c(F)c2)=O)CC2(CC2)C1 C(CC(C)C(=O)N(C(C)CNC(c1csc(Br)c1C)=O)C)OC CCCC(F)(F)C(=O)N(C)CC1CCCN1C(=O)COCC(C)(C)C n1(CC)nc(C(=O)N(C)CC2(CNC(C3CCSC3)=O)CC2)ccc1=O C1(C(=O)NCC2(F)CN(C(Cc3c(C)con3)=O)C2)C(C)(C)C1(C)C c1(C(N2CCN(CCC(=O)OC)CC2C)=O)c(O)nc2ccccc2c1C C1(CNC(C(n2ccc(C)n2)C)=O)CC(C)(C)CN1C(c1cccc(Cl)c1F)=O C1(CCC)CN(C(=O)C(C)C2CC2OC)CCN1C(=O)CCc1csnn1 N1(C(C(CC)=CCCC)=O)CC2CCN(C(=O)CC3(C)CCOCC3)CC(C2)C1 c1(C(=O)NCC(C)CNC(C2(Oc3ccccc3)CC2)=O)cc2c[nH]nc2s1 C(c1cncnc1O)=CC(=O)NC1CN(C(C2CCC(NC(C)=O)CC2)=O)C1 N1(C(C(C(CC)(C)C)O)=O)CC2(CCN(C(=O)C(C)CS(C)(=O)=O)CC2)C1 N1(C(C(COC)COC)=O)CCCCC1C(=O)NC(c1ncc(F)cn1)C c1(C(=O)NCC2C(NC(c3snc(O)c3Cl)=O)C2)cc2ccc(O)cc2[nH]1 C(CCCCC(=O)NCC(c1cnn(C)c1)O)N(C(=O)C(O)c1ccco1)C O=C1CC(CC(=O)NC2C3CC2N(C(c2cccs2)=O)C3)C(=O)N1 CN1CCC(C)(C(=O)NCC2CC3CC3N2C(c2cnn(C(C)(C)C)c2)=O)C1=O c1(OC)ccc(C2=NOC(C(C)C(N3CCC34CCOC4)=O)C2)cc1 C1(CNC(CSCc2nc(C)sc2)=O)CN(C)CCN1C(=O)CNS(C)(=O)=O C1(C(N2CCC(OC)C2)=O)CC2CCC1N(C(c1nc[nH]n1)=O)C2 Cc1onc(-c2ccsc2)c1C(=O)NCC1CCCCC1NC(=O)CC(C)(C)F CN(C)NC(=O)CCC(=O)N1CC(N(C(=O)C#CC2CCCOC2)C)C2(CC2)C1 C1(c2ccccc2)(C(=O)NCCN(C(=O)C(O)CN(C)C)CCOC)CC1(C)C C(=O)(CC(CNC(=O)OC(C)(C)C)Sc1cccc(Cl)c1)N(CCOC)C N1(C(Cc2nc(-c3ccc(C)cc3)sc2)=O)CCC(SCC2CCCCCC2)C(C)C1 C1(C(=O)NC2CCN(c3ccccn3)CC2)CC2CCC(C1)S2(=O)=O c1(NC(C(C2CC3CC3N2C(=O)OC(C)(C)C)C)=O)cccc(C(=O)O)c1 N#Cc1cnc(C(=O)NCCCNC2(c3ccc(C(F)(F)F)cn3)CC2)c(F)c1 CC1(C)CCCC(C(=O)N(CCCn2cc(C3(n4nccn4)CC3)nn2)C2CC2)C1 C1(NC(N2CCC(C(C(=O)OC)F)C2)=O)CC12CCC(F)(F)CC2 C#Cc1cc(F)c(C(=O)NCCC(C)(C)CNC(=O)CC2CN(C)C2)c(F)c1 c1(C(=O)NC2C(CC)N(C(c3nc(C)c(C)s3)=O)CC2)cc2occc2n1C c1(C(=O)NCC2CC(C)N(C(c3cccc(N)n3)=O)C2)cc2cc(Cl)cnc2o1 c1(C(C(=O)NCC)N(C2(c3ccccc3)CC2(C)C)C)cc(Cl)ncc1OCC N1(C(CC23CC(C)(OC2)C3)=O)CCCC2CN(C(C3OC(C)CC3C)=O)CC12 Cc1cncc(CN2CC3(CC3C(=O)NCc3ccc(F)cc3)C2)c1 c1(C(=O)NCC2CC(C)N(C(=O)Cn3cc(C4CC4)cn3)C2)ccc(Cl)cc1O C1(C)(CNC(CCOCCC)=O)CCC(NC(=O)CCCCOC)C1 Cc1n[nH]c(C)c1C(C)C(=O)NCC1(F)CC(CNC(C2CCC(C)CC2)=O)C1 N1(C(C)=O)CCCCC1CC(=O)N(CCNC(C1(C)CC(C)=NO1)=O)C(C)C C1(C(N2C3CN(C(c4ccncn4)=O)C(C3)C2)=O)COc2cc(Cl)ccc2C1 CCCS(=O)(=O)C(C)C(=O)N1CCC2(CCCN2C(C2CC(=C3CC3)C2)=O)C1 Cc1cc(C(=O)NC(C)(CNC(C2(CCF)CCC2)=O)CO)c2nccn2c1 N1(C(C2CCCSS2)=O)CC2=CC2=NC=CNCC(NC(C2(Cl)CC2)=O)C1 CC(C)C(CCN(C)C(c1cccc(C(N)=O)c1)=O)NC(c1cccc(F)n1)=O c1(NCCCC(C)NC(C2(C)C(C)(C)C2(C)C)=O)nnc2c(c1C#N)CCCC2 C1(CNC(C=CCNC(C(C)Cn2ccnc2)=O)=O)CCC=CCC1 C1(NC(C(C)CC(N)=O)=O)CCC(N=c2nc[nH]c3[nH]c(I)cc23)C1 C#CCC(CC#C)C(=O)N1CCCC(N(C(=O)C(Cl)Cl)C)C1 N1(C(=O)C(O)Cc2ccccc2)CCN(C(=O)CCc2cccc(Br)c2)CC1 C1(C(=O)Nc2c(C)cccc2O)C2CC(O)C(C2)N1C(C1(C)CCSCC1)=O C1(NC(c2ccc(C)nc2N)=O)CS(=O)(=O)CC1NC(=O)CSCCN(C)C N1(CCCC(=O)NCC(C)(C)CC2CC2)C(=O)NC2(CCCCCC2)C1=O C12(CC(=O)NCCC=CC=C)CCC1CN(C(c1cc(C)nc(C)c1)=O)C2 C(C(C)(C)C(F)F)NC(C1(C2N(C(CC(C)C)=O)CCC2)CC1)=O c1(OC)cc(OC)c(-c2cccc(CNCC3CCCc4ccccc43)n2)cc1OC C(C1CCN(C(c2cc(Cl)no2)=O)CC1)=CC(=O)NCC(C)(F)C(F)F c1(C(N(CCC#C)C2CC2)=O)sccc1CNC(C1CCCCO1)=O C1(=O)C2CC1Cn1ccnc12.Cn1ncc2cccc(N)c12.C(=O)O c1(C(=O)NCC(CCOC)NC(c2ccnc(C)c2)=O)cc(F)c(F)cc1F C(CCCCS(C)(=O)=O)NC(c1cncnc1C1CC1)c1n(CCCSC)nnn1 Cc1cc[nH]c(=N)c1C(=O)NCC12CC(NC(c3cc(O)nn3C)=O)(CO1)C2 Cc1ncsc1COCC(=O)NC1CC(C)(NC(c2cnn[nH]2)=O)C1 C1(NC(c2ncoc2C2CCCC2)=O)CN(C(c2cc(CO)on2)=O)CC1F N1(C(c2cc(C)c(C)s2)=O)CCC2C(CCN2C(=O)COc2ccccc2)C1 N1(C(C=CC)=O)CCCN(C(=O)COc2ccc(CC)cc2)C(CO)C1 C1(CCCNC(CCC)=O)CN(C(C2(C(N)=O)CC2)=O)CCO1 c1(CC(=O)NCC(CN(C(=O)CCc2ccc(O)cc2)C)O)cccc(C#N)c1 C=C1CC2CCCC(C1)N2C(=O)CCC1CCN(C(=O)CCCOC(C)=O)C1(C)C c1(C(=O)OCC)nnc2n1CCN(C(=O)NC(C)(CC(F)(F)F)c1ccncc1)C2 C1(CNC(C2CC(OCC)C2)=O)CCCC(NC(=O)COc2ccsn2)C1 C(=O)(C1=CCCC1(C)C)N1CC(C(C)NC(=O)NC2CC2)C1.C12CC(C1)C(=O)OC2 c1(NC(C2C(C(=O)NCc3csc(-c4ccccc4)c3)C2)=O)cc(Cl)cc(Br)n1 N1(C(Cc2c(C)ocn2)=O)CCN(C(c2ccc(O)nc2Cl)=O)C(CCO)C1 c1(C(N2CCC(Cc3nc(CC)no3)C2)CC)ccc(Br)cc1 c1(OC)ncc(C=CC(=O)NC2CCC2NC(=O)C(C(C)C)NC(N)=O)cn1 c1(C(=O)NCCC(C)(C)NC(C2CC3CC2C2CC32)=O)cnn2c1OCCC2 c1(C(N(CC(C)NC(C(CC)OCC)=O)C)=O)c(C)nn(C)c1Cl N1(C(C2C(c3cn(C)nc3)C2)=O)CCN(CCO)c2ccc(Cl)cc21 N1(C(C(C(C)CC)N(C(COCCC#C)=O)C)=O)CCC(C)C2(CCC2)C1 C1(NC(c2cc(CCNC(c3ccc(C)o3)=O)on2)=O)CC2(CCC2)C1O Cc1c(N)c(C(=O)NC2CC(NC(=O)CC3CC4(CC4)CO3)C2)cc(F)c1F c1(N2CC3C(NC(CCCOCCC)=O)C3C2)ncnc2c1nnn2C(C)C CN1CCCCC1CC(=O)NCc1cccc(C(N2CCC(F)CC2)=O)n1 c1(CC(N2CC(NC(CCCNC(=O)OCC)=O)C(C)C2)=O)ccc(F)c(F)c1 c1(C(N2CCC(N(C)C(c3cnc(C4CC4)s3)=O)C2)=O)occ2c1CCOC2 C1(NC(=O)C=Cc2cccs2)CN(C(=O)Cc2ccccc2)CC2CC12 c1(C(=O)NCC2CCCCCN2C(=O)Cc2nc[nH]n2)csc2c1CCCC2 c1(C(=O)NCC2(C(N3C(C(C)C)CCCC3)=O)CCC2)cc[nH]c(=N)c1Cl c1(NCc2c(F)cncc2)[nH]c(=NC2CC3CC2CC32CC2)nc2sccc12 C(CC(C(C)(C)C)NC(c1c[nH]nc1-c1cccs1)=O)N(C(=O)C1=CCOC1)C C(C(C)(O)CC(=O)NC(C)(C)CCC1CCN(C(c2coc(C)n2)=O)CC1)OC CC1CC(Nc2cccc(-c3ccccc3)c2)CCN1C O=S(=O)(c1ccc(NC2(c3ccccc3Br)CCC2)nc1)NCCCCCO c1(NC2CCCO2)cc(C(C(=O)NC(C)C2CC2)N(CC(C)C#N)C)ccc1F CCC(C(=O)NCC1CC(NC(c2c(C(C)C)cccc2C)=O)C1)C(C)C C(CC(=O)NCC(CO)NCc1cc(O)ccc1O)(C(F)F)NC(=O)OC(C)(C)C N1(C(CC)=O)CCCC1C(C)C(=O)NC1CCN(c2ccncc2)C1 C1(C(=O)NC(C2N(C(CN(C(C)C)C)=O)CCC2)(C)C)(CSC)CC(C)(C)C1 c1(OCC)cc(Br)ccc1Cn1cc(C(C)NS(=O)(=O)CCCCCl)cn1 N1(C(c2c(CC)cccn2)=O)CCN(Cc2c[nH]c3ccncc23)CC1(C)C N1(C(CC(CC)NC(=O)C(O)C2CCCC2)=O)CCc2nncn2CC1 Cc1oc(C#N)cc1C(=O)NCC(O)CNC(=O)Cc1ccc(O)nc1 C(c1ccc(F)c(F)c1)=C(C(=O)NC(CCN(C(C1(CC)CCC1)=O)C)C)C C1(N(C(c2ccc(CSC)o2)=O)C)CN(C(=O)Cc2ccncc2)CCC1O CCC(C)C(O)C(=O)NCC1(F)CCN(C(c2ccc(-c3ccon3)cc2)=O)C1 C1(CCNC(c2n(CC=C)ccc2)=O)CCN(C(C2CCCCC2OC)=O)CC1 N1(C(C(CNC(C)=O)(C)C)=O)CC=C(C(=O)N2CCOCC(CO)C2)C1 c1(C(F)(F)F)nc(NCCCc2ncc(Br)cn2)cc(=NC2CC(=C3CC3)C2)[nH]1 C=CCCCCC(=O)NC1(CC)CCCN(C(c2ccc(CC3CC3)s2)=O)C1 CCC(C(C)(F)F)C1CCN(C(=O)NCC)CC1.C1(CC)CN1CC N1(C(c2ccc(OC)s2)=O)CCC(O)(CCNC(c2nnc(O)nc2O)=O)CC1 c1(OC)ccc2[nH]c(C)c(C(=O)NC3CN(C(=O)C(C)(CO)OC)CC3C)c2c1 c1(C(=O)NC(CNC(c2cc(OC)n(C)n2)=O)(C)C(C)C)cc(O)nc(O)n1 Cc1onc(C(=O)N(C2CCC(n3cc(CCOC4CCC4)nn3)CC2)C)c1F c1(OCC)cnc(N2CCC(NC(=O)CCC3CCOC3)CC2)nc1C C12(CNC(=O)C3=C(Cl)CC3)CCC(CNC(=O)CC3C=CCC3)(CC1)CO2 c1(OC)ccnc(COC(c2cc(CO)oc2C)=O)c1C C1(NC(C2CC(=O)NC2)=O)CCC2(CC1)CN(C(C1(CCF)CC1)=O)C2 c1(C(=O)OC)ccc(C(=O)N(CC(O)CN(C(C2COCCO2)=O)C2CC2)C)nc1 C(CC(C(=O)N(C)CCNC(=O)CS)N(C)C)SC.c1(C2CC2)ccccc1F c1(OC)c(Cl)cc(O)c(Cl)c1C(=O)NC1CCCC1NC(C1CC12CC2)=O C1(CNC(C(C2CCN(C(c3ccn(C)c3)=O)C2)(C)C)=O)CCC(=O)NC1 c1(C(C(F)(F)F)NC(=O)NC2(c3ccccc3Cl)CC2)ccc(Cl)cc1 C1(CC(=O)NCC(=O)OCCCC)CCCCN1C(C1CCOC(C)C1)=O C1(C(=O)NCCOC2CCN(C(CC=C)=O)C2)CC2(CC(=O)N2)C1 C(=O)(CC1CCOc2ccccc21)NC(C)CCCNC(C1CCCCN1C)=O C1(C(=O)NCC#CC(N2CCC(C(C)(C)O)CC2)=O)(CC)CCOCC1 c1(NCC(C)(C)OCC)[nH]c(=NCC2(C)CCC(C)CC2)nc2c1cnn2C c1(C(N(CCCNC(CC(CC=C)(C)C)=O)CC)=O)oc2c(C)cccc2c1C C1(CNC(c2ccco2)=O)CC2(CCN(C(=O)CC3CC3C(F)(F)F)CC2)CO1 c1(OC)ccc(S(=O)(=O)NC2CN(c3nc(C(F)F)no3)C2)cc1C(N)=O C1(C(=O)NC(CC(=O)N(C2CCCC2)CC)C)C2CN(CC3CCC3CSC)CC12 C1(NC(C(C(C)C)NC(C)=O)=O)CCC2CCN(C(c3ncnn3C)=O)C1C2 CC(C)CC(O)C(=O)N1CCCC(NC(=O)Cc2ccsc2)C1 C1(C2N(C(CNC(c3c(C(=O)NC)csc3)=O)=O)CCC2)CCN(C(C)=O)CC1 N1(C(CNC(c2c(C)ccn2C)=O)=O)CC2(CCC(O)CC2)C1 Cc1nc2c([nH]1)CN(C(=O)CN(C(=O)CCCC1CC1)C1CCC1)CC2 N1(C(Cc2ccn(C(C)C)n2)=O)CC2CC2(NC(c2cc(Br)cs2)=O)C1 c1(OC)c(C)cc(NC(C2CN(CC3CCCC(C)C3)C2)=O)cc1Br N1(C(c2c(N)snn2)=O)C2CCC1CC(C(=O)NC1CCCC(C3CC3)C1)C2 c1(SCC(N2C(C(C)NC(C3CCC(CO)O3)=O)CCC2)=O)cccc(C#N)c1 C1(N(C(CN(C)CCc2ccccc2)=O)C)CN(C(c2ccsn2)=O)CC1(C)C C=CC(CCC)CC(=O)N1CC(NC(=O)C=COCC)CC1C N1(C(c2c(C)ncs2)=O)CC(NC(c2csc3cccnc23)=O)C(C2CC2)C1 C(=O)(CCCCC(N)=O)NC(C(C)NC(c1cc(OC)c(O)cc1)=O)C n1(CC=C)c(N(C)C(c2cnnn2C)C)nnc1-c1n[nH]c(=N)[nH]1 O=C(CCCCc1cccs1)NC1(CO)CCN(C(=O)CCC2CCCOC2)C1 C(CC(C(C)C)NC(=O)C(Cn1cccn1)NC(=O)C(N)=O)OCC C1(O)(C(=O)N(C)CC2CCN(CC(C)C)C2)CCN(C(=O)NC2CCCO2)CC1 C1(C(N2CC(NC(CC3(C)CCC3)=O)C2)=O)Cc2ccc(F)cc2C1 C1(O)(CN(C)C(C2(C(N)=O)CCCC2)=O)CCN(C(c2cnc(Cl)[nH]2)=O)C1 c1(NC(C)CCF)nc(N2CC3CCC(C2)C3(F)F)nc2sccc12 CCCCC(O)C(C)C(=O)NC1CN(C(=O)CCn2cnnn2)CC2CC12 C1(CCO)(NC(C(n2cc(CCS(=O)(=O)N(C)C)nn2)C)=O)CCCSC1 CC1CN(C(C23CCCN(CC2)C3)=O)CC(C)N(c2ccc3nnnn3n2)C1 C1(CNC(C2CC=CCC2)=O)CC2COCC2N1C(c1occ2c1CCC2)=O c1(C(=O)NC2(CNC(C(CCSC)O)=O)CCCC2)ccc2snnc2c1 CCCC(CC1CCCC1)C(=O)N1CCCC1CN(C)C(C1(C(F)(F)F)CC1)=O C(=O)(C(F)(CNC(C1CC12CCCCC2)=O)C(C)C)NCc1c(C)n(C)nc1 C1(CN(C(C2(CC(=O)OC)CCC2)=O)CC)CCCN1C(=O)C(C)=C1CCC1 N1(C(CC(CC)(F)F)=O)CCC2CN(C(c3ccc(C4CC4)cn3)=O)CCC2C1 c1(NCC(CNC(C(CCC)OCC)=O)O)cc2nc(O)oc2cc1[N+](=O)[O-] C1(C(N2CC(CNC(C(C(C)OC)N(C)C)=O)C2)=O)CC2(CCC(F)(F)CC2)C1 C1(C(N2C(CNC(Cc3c(OCC)cccc3)=O)C=CC2)=O)CCCCC12CC2 N1(C(c2nnc(C(F)(F)F)s2)=O)CC2CC2(C(=O)NCCn2ccnc2)C1 C(C(C(=O)C(CSCC)=O)OC)N.C(C)(C)(COC)N CCCCC(CC(=O)N1CC(C)(C)C12CCC2)NC(c1ccnn1C1CC1)=O C1(CNC(N(c2ccccc2)C(CC)(C)C)=O)CCCC(NC)CC1 C1(CCCNC(=O)Cc2ccccc2)(CNC(C2C(OCC)C2)=O)CCCC1 N1(C(c2cc(F)c(Cl)cc2F)=O)CCC2CN(S(=O)(=O)c3cnc[nH]3)CC2C1 c1(N2CCCC(CC)(CC)C2)nc(NCC(C(F)(F)F)OC)c2cnn(C)c2n1 CC1CCc2c(sc(NC(C3CN(C(=O)CN4CCNC4=N)CC3C)=O)c2C#N)C1 CN1C(=O)NCC1C(N1CCC(CC23CC(CCn4cncn4)(C2)C3)CC1)=O N1(C(c2c(COC)cc[nH]2)=O)CCOCC1CN(C(=O)CC1CC(OC)C1)C c1(C(C)NC2(c3n(CC)nnn3)CCN(CC)CC2)ccc(S(C)=O)cc1 O=C(CCCCc1ccccc1)NCC1(CNC(=O)CC2CC3CC3C2)CC1 c1(C(N)=O)ccc(S(=O)(=O)N2CCN3CC23)nc1.C(N)=O CC1(C(=O)NCc2csc(C(N3CC4C(C(N)=O)C4C3)=O)c2)SCCCS1 c1(N2CCC(C)OCC2)ccc(S(=O)(=O)NCC(O)CCC2CC2)cc1Br C(=O)(C#Cc1ccccc1F)NC(c1ccc(OCCC)c(OC)c1)C n1(CC(N2CC(CCNC(C(CSC)C)=O)C2)=O)ncc(C#N)c1N C(=O)(CC(CC)C(F)F)N1C(CNC(CNS(CCOCC)(=O)=O)=O)CC(O)C1 CCCC(C)C(=O)N1CCC(CN(C(=O)Cc2nn(C)cc2Cl)C)C1 c1(C(N2CC(O)(CNC(C=COCC)=O)C2)=O)[nH]c(Cl)c(Cl)c1Br CN1CCCCC1Cc1nc(Cn2cncn2)nn1-c1ccccc1 C1(NC(C(c2cc(C)cc(C)c2)C)=O)CCC2CCN(C(=O)CC34CC(C3)C4)C12 c1(C(N2CC(CCNC(C=NOC)=O)S(=O)(=O)CC2)=O)cc(F)c(F)c(C#N)c1 c1(NCC2(F)CC(NC(C3(C(N)=O)CC3)=O)C2)ccc([N+](=O)[O-])cc1F N1(C(c2cc(OC)c(C(F)(F)F)cc2)=O)CCCN(C(C2CCCO2)=O)CCC1 C(=O)(CC(O)CC(C)(C)C)N(CC(C)O)Cc1cccnc1.C1(=O)CN1 Cc1oc2ncnc(O)c2c1C(=O)NC1CN(C(C2CCCC(C)(C)CC2)=O)C1 c1(NC(C(=O)NC(c2ccccc2OCC)CC(=O)OC)=O)ccc(C)c(CN)c1 N1(CC(=O)NCCC2CCC(NC(CSc3nc(C)[nH]n3)=O)C2)CCCS1(=O)=O C1(NC(=O)NCc2ccccc2)CCN(Cc2nnc(C3CC3)s2)C2(CCC2)C1 CC(C)C(C)(CO)NC(=O)C(O)CNC(=O)C=CC(F)F N1(C(=O)CSC2CC2)CCC(C2CCN(C(c3ccc(F)s3)=O)C2)C1 C#CC1(F)CN(C(=O)CC2CCN2C(=O)CCC(=O)NC2CCCCC2)C1 CC1(C)CC(C(N2CC(CO)(NC(c3cnns3)=O)C2)=O)CO1 Cc1nn(C)c(C)c1C1C(CNC(=O)NCCC(C)CO)CC(=O)N1C C1(C(=O)NC(C)(C)C(N)=O)CCCC(NC(=O)Cc2ccccc2F)C1 C(=O)(CC(C)C(C)C)NC(C)=O.c12ccccc1NCC1CCN2C1 c1(C(=O)NCC2(CNC(c3c(Cl)cc(C)s3)=O)CC2)ccc2nccn2c1 CC(CC(C)NC(=O)C(c1ccc(Br)s1)=O)NC(C1CCCS1)=O c1(C(C2(CC)COC2)NCCSc2nnnn2C(C)C(=O)OC)coc(C)n1 N1(C(COCc2cc(C)on2)=O)CC=C(CNC(C2C3CC3C3CC23)=O)CC1 c1(C(C(=O)NCCC(CC)O)N(C)C)cccc(Br)c1 C(CCCC(=O)N1CCCC1(C)C(=O)NC1CC=CCC1C)NC(C)=O N1(C(c2c(C)ccs2)=O)CCC2CCC(C1)N2C(c1cn(C2CCOC2)nn1)=O c1(C(=O)NC2CC(NC(C3CCCC(OC)C3)=O)C2)cc(S(N)(=O)=O)cnc1C N1(C(c2nnc(CC)s2)=O)CC2CCC(C1)N(C(=O)CCS(C)(=O)=O)C2 C(=O)(CCC1=CCCCC1)NC(C(C)C)(C)CNC(=O)C(C)Cc1cnn(C)c1 Nc1c(C(N2CC(NC(=O)Cc3ccco3)C(CO)C2)=O)cccc1Br c1(C(N2C(CNC(Cc3cnc(C)[nH]3)=O)CC(F)C2)=O)cc(C)nc(O)n1 CCCCC(CNC(=O)C(C1CCOC1)OCC)NC(=O)CC1CCOC1C CCCC(C)CC(=O)NOC(CC(C)C)C(=O)NCC12CC(F)(C1)C2 c1(SC)cncc(C(=O)NC2CC(C(C)NC(C3(n4cccn4)CCC3)=O)C2)c1 C(=O)(CS(=O)(=O)C1CC1)NCC1N(C(CCCC(=C)C)=O)CCOC1 C1(CNC(CCSCCC)=O)CCCC1C(N1CC(NC2CCC2)C1)=O C(C(=O)NCC(O)CNC(c1sc(C)c(Br)c1C)=O)(C(C)(C)C)OC C#CCCCC(C)C(=O)NCCCCC(C)NC(=O)C(c1ccc(Cl)nc1)(F)F C1(C(=O)NCC=CCNC(CCCc2cc(C)no2)=O)CCC(=O)N(C(C)C)C1 c1(OCC)cc(C(N2CC(C)(NC(C3CCN(CCC(C)C)C3)=O)C2)=O)sn1 c1(C(N(CCC(C)NC(=O)C(F)=CCCF)C)=O)nc2ncc(Br)cn2n1 C(CCCC(=O)NCC(CO)NC(=O)Cc1cncnc1O)OCC C1(N(C(=O)CSc2ccccn2)CC)CCN(C(c2ccnn2C)=O)CC1 C1(CC)CC(C(N2CCC2CC2CCCC2)=O)CCN1C(C1CC1(F)Cl)=O c1(NC(C2CC(F)CN2C(C2CCCS2)=O)=O)ccn2nccc2n1 C(=O)(CC(C(F)F)n1ccnc1)NCC(C)CNC(c1ocnc1C1CC1)=O C=CCCC(C(=O)Nn1cnnc1C)NC(=O)CN(C(=O)C(C)C)C Cc1cc(O)ncc1C(N1CCCC(C(C)NC(=O)CCc2ccncc2)C1)=O c1(C2C(SCCC(N3CC(CCNC(c4cc[nH]n4)=O)C3)=O)C2)ccccn1 C1(NC(C(C)OC)=O)CN(C(=O)Cn2ccnc2C(C)C)CC1C(F)(F)F C1(CNC(C(CC)F)=O)CN(C(C2CC2C)=O)CC1(F)CO S(=O)(=O)(c1ccc(C(N2CC(NC(c3cc(OC)no3)=O)C(O)C2)=O)cn1)NC c1(C(N2CC3CN(C(C45CC6CC4C5C6)=O)CC3C2)=O)ccc2nc[nH]c2n1 c1(OC)c(C(=O)NCC2CN(C(=O)C(C)(C)CO)CCC2(C)C)nc(O)nc1O CCC(CCCC(=O)Nc1cc(C)nnc1C)NCC1CC1.C(C)(CO)C1CC1 C1(NC(CSc2c(C)ocn2)=O)CCCN(C(=O)CN2CCCOC2=O)C1 CC1OCCC2CCCN(C(=O)NCC3CCC(C(C)(C)C)CC3)C2C1 c1(C(=O)NCCC2N(C(c3c(SC)snn3)=O)CCSC2)ccc([N+](=O)[O-])cc1 c1(NC(=O)NC(C(C)O)C)nc2c(s1)COCC2 N1(C(CCCCN(C(C2C(COC)CCO2)=O)C)=O)CCc2ccccc2C1 C#CCC(C)OC(=O)CCN(CC(C)SC)CC c12cc(OC)cc(c1)C(=O)O2.c1(C(=O)OC)ccccc1NS(C)(=O)=O c1(C(=O)NCC2C3CN(C(C4(C)CC4(F)Cl)=O)C2C3)cnc2c(F)cccn12 Cc1cc(NC(c2cc(F)ccc2O)=O)ccc1NC(C1OCCN(C)C1=O)=O c1(C(N2CC(N(C(=O)C=Cc3cocn3)C)C(F)C2)=O)cnc2c(c1)COCC2 Cc1nn(C)c2c(N(C)Cc3ccncc3F)nc(=NCc3ccccn3)[nH]c12 c1(C(=O)NCC(O)CNC(c2sccc2C(F)F)=O)cc(O)nc2c1CCCC2 C1(CCNC(=O)Cc2ccnn2C2CCCC2)CN(C(C2CC2CF)=O)CCO1 c1(C(N(CCCNC(=O)CCCc2nc(C)cs2)CC)=O)cc(C(C)C)oc1C C1(OC(CC)C)CCCCC1C(=O)NCCCOC C1(CN(C)C)CCN(CC(O)COC2CCOCC2)C1.c12cnn(c1)C2 C(=O)(C(F)CCCC)NC1(CC=C)CN(C(c2cncc(C(F)F)c2)=O)C1 C(=O)(C1=C(C)OCCC1)N1C(CNC(=O)CNC=O)CC(OC)C1 C1(C(=O)NC(C)(C)C)CC2CCC1(Nc1cnc(-c3nn[nH]n3)cn1)C2 c1(C2(CN=C(NC3C(C=C)C3)NC3CCCC3)CC2)ccc(Br)cc1F C(=O)(C1CCCn2nccc21)N1CCCCC(NC(c2c(C)cnnc2O)=O)C1 C1(C2(N3CCCC(C4(C)COC(=O)N4)C3)CC2)CN=C(c2ccccc2)N1 C1(C(=O)NCC2OCCN(C(C)C)C2)CC12CCN(C(=O)C(C)(C)O)CC2 c1(CC)ccc(OC(C2C(C(=O)OC)CCCC2)=O)c2[nH]ccc12 CC1=NOC(CCNC(C2(NC(=O)CSc3ccccn3)CC2C)=O)C1 C1(C(N(CCOCC)C)=O)CC12CCC2.C12(COC1)CC(=O)NCCN(C)C2=O c1(COC)cccc(CC(=O)NC(C)CCCNC(=O)Cn2cc(CO)nn2)c1 C=CCCCC(C)CC(=O)N1CC2(C1)SCCC2NC(c1cc[nH]c1C1CC1)=O c1(C(N2CCCC2CC2CCCC2)C(=O)NCC=C)ccc(C(C)CC)cc1 C1(C2CCN(C(C(C)=CC)=O)C2)CCCCN1C(c1cc(C)[nH]n1)=O c1(CC)ncoc1C(=O)NC1(CNC(=O)CCCOc2cccnc2)CC1 CC1CN(C(=O)CC2(O)CCC2)CC1CC(=O)Nc1cnsc1 N1(C(CNC(CN(C(CNC(CCC)=O)=O)C(C)C)=O)C)CCOC(C)C1 c1(C(=O)NCCCN(C(=O)C(C)(C)C(N)=O)C)nccn2c(Br)cnc12 c1(C(=O)OC)ccc(COC(c2cnnc(I)c2)=O)cc1 C1(NC(=O)COCC2CC2(Cl)Cl)CC2(C1)CC(NC(=O)CC1CC(C(=O)O)C1)C2 C1(CNC(C2C(C(=O)OC)C2)=O)N(C(C2CCC3(CC2)CC3)=O)CCCC1(C)C Cc1cc(CCC(=O)NC(C)CCNC(C2CC(=C3CCC3)C2)=O)cc(C)c1 CC(F)CC(=O)N(C1CC1)CC1(CC(=O)NCC2CCCOC2)CCCC1 c1(CNc2ccc(C)c(Cl)c2F)ccc2c(c1)OCCCO2 CCC(C(=O)NCCC(C)(C)NC(=O)Cc1sccc1C)NC(C)=O N#Cc1ccc(F)c(C(=O)NC2C=CC(C(=O)NCc3noc(C(F)F)n3)C2)c1 c1(OC)cc[n+]([O-])c(C(=O)NC23CC2CN(C(c2ocnc2C)=O)C3)c1 Cn1cc(-c2cc(C(N3CCC(NC(=O)C(c4cccnc4)=O)C3)=O)on2)cn1 N1(C(c2cc(COC)no2)=O)CCC2(CC1)CC2(C)C(=O)N(C)CC1CCC1 N1(c2nnc(-c3ccc(C)cc3C)n2CC(C)C)CC(CO)C(C)CC1C C1(C(=O)NCC2N(C(C(C)C3CCCO3)=O)CC2)(CF)CC2(CCC2)C1 c1(C2N(C(c3ncnn3C)C(=O)NC(C)C)CCC2)cccc(F)c1 c1(C(N(CCCNC(C(CC)C(C)C)=O)CC)=O)ccc([N+](=O)[O-])cc1C N1(C(Cn2c(C)nc(C)n2)=O)CC(NC(c2[nH]cnc2C)=O)C2CC2C1 n1(CCC)nc(CC(C)C)nc1-c1csc(C)n1 c1(CCC(=O)NC2CC(C(=O)NCc3nc(CC)on3)C2)ccc(Cl)c(Cl)c1 N1(C(CCCC=C)=O)CC2(CCN(C(=O)C(O)C(C)CC)CC2)C2COCC12 C=CCCCC(C(=O)NCCCCCCF)NC(C1CCO1)=O c1(C(N(C2CCN(C(=O)CCC3CCCCCC3)C2)C)=O)ccn2ncccc12 Cc1nc2[nH]c(C(=O)NCCCN(C)C(c3ccc(C4CC4)nn3)=O)cc2s1 C(N=c1[nH]cnc2cccnc12)C1C(CNC(CC(C)(O)C(F)(F)F)=O)CCC1 N#Cc1ccccc1CNC(C1CCN(C(=O)Cn2cnnc2)CC1O)=O N1(C(CCCCC#C)=O)CC2(C1)SCCC2NC(C1CC1OC)=O Cc1nc(N2CCN(C(C3CC3(C)C)=O)CC2)nc2c1CCCC2 Cc1ccccc1CC(N1CCNC(C(=O)Nc2[nH]cnc2C#N)C1)=O CCCC(C)(CCC)C(=O)N1CCN(CCN(C)C(C2C3CCCC23)=O)CC1 N1(C(C2(CC)COC2)=O)CCCC(C)(C(N2CCC(C(C)(C)O)CC2)=O)C1 Cc1ccc(CC(=O)NC(C)CC(C)NC(=O)Cc2occc2C)s1 Cc1ccc(C(N2CC3CC2C3NC(=O)COCc2cccnc2)=O)c(N)c1 C1(C(N2CC3C(NC(C(C)OCC#C)=O)C(C3)C2)=O)C2CCCCCCC12 c1(OC)ccc(CNC(=O)C(N2CCCC2c2cccc(Cl)c2)=O)cc1 C1(CCNC(C2(C=C)CCC2)=O)CN(C(=O)Cc2[nH]cnc2C)CCCO1 C1(C(=O)OC)(N(C(C2CCCC(C(F)(F)F)C2)=O)C2CC2)CC2CC1C2 N1(C(c2cc(C#C)cc(N)c2)=O)CC(C)(C)OCC1CNC(C1CC1F)=O c1(C(N2C(CN(C(=O)Cn3cc(CO)nn3)C)CCC2)=O)cc2c([nH]1)CCC2 N1(C(CN(C2CC(C#N)C2)C(C=CCCC)=O)=O)CCC(O)(CN(C)C)C1 C1(CC)CC(C(=O)N(CCNC(=O)C(=O)NCC(F)(F)F)CC2CC2)CCO1 c1(CC(C)C)ncc(C(=O)N)[nH]1.C(=O)(C(F)C1CCOC1)CCNCCCN(C)C Cc1ncc(C(C(=O)NC2CCOC2)N(C)C(C)C2CC2)cn1 N1(C(CC(CC)C2CC2)=O)CCOC(C)C1C(=O)Nc1cc(F)ccc1O C1(C)(CNC(C2(OCC)CC2)=O)CCCN1C(c1coc(Cl)n1)=O c1(C(=O)NC2C(NC(Cc3cc(C)sc3)=O)C2)cc(Br)c(C)cc1F C#Cc1ccc(C(=O)NCCCNC(=O)CC2CCc3cnn(C)c3C2)cc1C C1(C(N2CC(O)(C(C(N3CCC(CC)(CO)C3)=O)F)C2)=O)OCCCC1(C)C C(C)(C)(CCCNC(=O)COc1cccc(F)n1)NC(C(CC)=CC)=O CCC(CC)(CCNC(=O)CC1CC1)NC(=O)Cc1occc1C CN1CC2(CN(C(C3(NC(c4cnc(C(=O)N(C)C)o4)=O)CCC3)=O)C2)C1 C1(C(=O)NC(c2ccccn2)C)CC2CCCC2N1C(=O)Cc1cncn1C C1(C(=O)NCC2CN(C(CCN(C(CCC)C)C)=O)C2)CCN(CC(F)(F)F)C1 c1(SCC)nc(-c2ccc(C3CC3)cn2)n(C2CCC(C)(C)C2)n1 c1(CN(CCC)C(c2cccc(Br)c2)c2ccncc2)ccccc1Cl CCC(O)C(C)(C)C(=O)N1CCC(CCOC)(NC(=O)CC2CC=CC2)CC1 c1(C(c2nnnn2C2COC2)NCC(C)CO)ccn(C(F)F)n1 CCCC(CCC)C(=O)N1CCC(NC(C2CC3(CCOCC3)C2)=O)C(F)C1 Cn1c(C(=O)NCC2(O)CCCN(C(C3(C)CSC3)=O)C2)cc2ccsc12 N1(C(c2c(CNC(c3cc(CC)ncn3)=O)ccs2)=O)CCC(C)CC1C(C)C c1(C(=O)NC(CNC(C2CCC(C(C)C)CC2)=O)(C)CO)cc(Cl)c(F)c(Cl)c1 c1(C(=O)NCC(N2CCN(C(CCCOC)=O)CC2)=O)cccc(C)c1Br c1(C(=O)NC(CNC(c2cccc(Cl)c2F)=O)C2CCC2)cccc2[nH]ccc12 N1(C(CC2C(C)(C)C2)=O)CCC2(CC1)CCN(C(C1CS(=O)(=O)C1)=O)C2 c1(NC(C(C=CC)O)=O)ccc(Cl)c(C(=O)OC)c1.C1(=O)CCN1 C1(NC(COCC(=C)C)=O)COC2C(NC(c3nnsc3C(F)F)=O)COC12 C(=O)(C1=CS(=O)(=O)CCC1)NC(C(C(C)C)NC(c1ccc(C(N)=O)o1)=O)C C(C(C(F)(F)F)N1CCN(C(c2cncnc2)=O)CC1)NC(C1CC(C)(C)C1)=O C#CCC(CC#C)NC(=O)CC1(NC(=O)C(C)(C)F)CC1 c1(C(=O)NC2CC(NC(C(C)OCC(F)(F)F)=O)CC2O)nc2c([nH]1)CCCC2 C1(C(=O)NC2C(C)(C(F)F)C2)CCCN(C(c2cn(C3CC3)nn2)=O)CC1 C(CC(CO)C(C)C)NC(C(C1CCC1)NC(c1c(CC)ncnc1)=O)=O c1(NC(C(=O)N(C)CC2C(C)C2)=O)cnn(-c2ccncc2)c1C(F)F O=C1CCC2(CCN(C(=O)NCC3C4CCC3N(Cc3ccccc3)C4)C2)N1 c1(C(N2CCC(NCC(C)C)CC2)C(=O)NC)cc(OC2CCC2)ncc1Br C1(CNC(c2c(C(C)C)ocn2)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC1C C1(NC(c2c(OC)nc(C)cc2)=O)CCSC12CN(C(=O)C=CCN(C)CC)C2 C(=O)(CCCCCCCS(C)(=O)=O)NC(CC)CNC(C1CCN(OC)CC1)=O N1(CCCNC(N2CCC(NC(C3(CCOC)CC3)=O)C2)=O)CCC(C)(C)C1 C1(C(N2CC(CCNC(CCc3cccc(C)c3)=O)C2)=O)CCCC(C#N)C1 O=C(N=c1[nH]oc2ccc(F)cc12)C1CCCN1c1ncccn1 c1(C(=O)NC2CCC(NC(C3(CC4CC4)CCC3)=O)C2)cc2c(o1)CCCC2 CC(CCC(F)(F)F)NC(C1CC(F)CN(C(=O)CN2CCN(C)CC2)C1)=O N1(C(c2ccc(C3CC3Cl)s2)C(=O)NCC2CC2)CC2CC3CC(C2)CC1C3 C1(O)(C(C)(C)C)CCN(C(=NCCCCCN2CCCC2)NC2CCC2)CC1 O(NC(=O)C#CC1CC1)CC(=O)NCCCCCC#C C1(C(NOCCC=C)=O)CCN(C(=O)CC(O)C(C)C)CCO1 C1(C(N2CC3C(NC(c4ccc(COC)[nH]4)=O)(C3)C2)=O)CCc2[nH]nc(O)c2C1 C1(C(N2CCC(CNC(CC3CC(=C)C3)=O)C2)=O)(COC)CCCC1O C1(CN=C(NC2(C)CN(C(C)=O)C2)NCc2cnc(C)o2)OCC2CCC1C2.C(CO)O C=C1CCC1C(=O)NCCC(C)NC(=O)C(C)N(C)C C(=O)(C(O)CC[S+](C)C)NC1C(NC(C(c2ccccc2Cl)C)=O)CCC1 c1(NC(C2N(C(c3cc(OC)n(C)n3)=O)CCOC2)=O)cc(F)ccc1[N+](=O)[O-] Cc1ncc2ccc(C(N3CCCC(O)(CNC(=O)CCC4(C)CC4)C3)=O)cn12 c1(CNC(C(N2CC(C)C2)C)=O)cn(C2CCN(C(c3ccc(Cl)o3)=O)C2)nn1 CC(C)CCN(C1CCCO1)CCNC(N1C=C(C(C)NC(=O)OC(C)(C)C)C1)=O C1(C(=O)NCC(C)N(C(=O)C=C2CCC2)C)(CO)CCCC1 C1(C(=O)NCCC2(O)CCN(C(c3c(C)occ3)=O)C2)CCCCC(F)(F)C1 c1(C(=O)NC23CCC(C2)N(C(c2cncnc2)=O)C3)cc(Cl)cc2ccccc12 C12(NC(c3ccc(C)cn3)=O)CCCC1CN(C(C13COC(CF)(C1)C3)=O)C2 C(C1=NOC2CN(C(=O)C3=C(Cl)CCC3)CC12)NC(c1cc2nc[nH]c2cn1)=O Cc1nc(C)c(CN(C(=O)C(=O)NCC2(C)CC(F)(F)C2)C)s1 c1(C(=O)NC2CCN(C(CCCC=C)=O)C2C)ccc2nc(O)oc2c1 c1(COC)cc(C(=O)NCC(C)CNC(C2CC2c2ccc(C)s2)=O)no1 C1(C(N(CCCC)CC)=O)CN(C(=O)C(F)C(C)(F)F)CC12CCC2 C(c1ccc(F)c(Br)c1)=CC(N1C2C(NC(C3CCCCC3)=O)C(C2)C1)=O C1(C(=O)OCC)CN(C(C2(C)CC2C)=O)CC1F.n12nccc1NC(=O)C2.C(C)N Cc1nn(CC(=O)NCC2CCCN(C(=O)CCCN(C)C)C2)c(C)c1C=NO c1(C(N2CCC(C)(CNC(CCCCC)=O)C2)=O)cc(Br)cc(Cl)c1C CC1(C)CCN(C(c2ccc3nc[nH]c3n2)=O)CC1CNC(C1COC(=O)N1)=O C(C(C)(C)CC(=O)N1CCC(CNC(C2CCCN2N=O)=O)C1(C)C)OC C1(O)(C(C)NC(C2CCC(O)C2)=O)CCN(C(C2CN3CCN2CC3)=O)CC1 N1(C(CCc2ccc(OC)c(C)c2)=O)CC2(COC(CNC(=O)C(C)SC)C2)C1 C(=O)(CCCCC(=O)N=C1CCN(c2cccc(C(=O)OC)c2)N(C)C1)OC C(N=c1cc(-c2ccccc2)n(C)[nH]1)C12CC(C1)NC2.c1(CC)noc(CO)n1 c1(C(N2CC3C(NC(C(C)C(F)F)=O)C3C2)=O)cnc2c(c1)CCS(=O)(=O)C2 c1(C(=O)NC2C(NC(c3cncc(F)c3)=O)CCCC2)oc2ccccc2c1Cl C(C(C)(C)C(=O)N1CCCC1CN(C)C(c1cccn1C)=O)N(C)C C1(C(=O)NCc2ncoc2CNC(C(C)CSC(F)(F)F)=O)CCOC(=O)CC1 N1(C(CCc2cc(OC)cc(F)c2)=O)CCCC2(CNC(=O)C2)C1 C1(C(=O)NC2(CNC(C34CC(C)C3C4)=O)CC2)CCN(CCF)CC1 c1(NC(C2CC(C(=O)OC)C2)=O)ccc(S(=O)(=O)Nc2ccccc2Br)cc1 N1(C(c2ccc(C)c(CN)c2)=O)CCCC2(C1)C(=O)N(C)c1cccnc12 n1(C2CN(C(CN(C)CCO)=O)C2)cc(C)nn1.C12(C(=O)NC(C)C3CC3)COCC1C2 N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)C=C2CCCCC2)C(CC(=O)NC)C1 CC(C)CC(F)C(=O)NC12CC1CN(C(=O)C1=COCCC1)C2 N1(C(C2N(C(=O)OC)CCC2)=O)CCCC12CCN(C(=O)Cc1cc[nH]n1)C2 CC(C)(C)C(C)(C)C(=O)NCC1CCN(C(=O)CC2(C)CC2(F)Cl)C1 c1(C(N(CCNC(Cc2c(C)n(C)cn2)=O)CC2CC2)=O)cnc(O)c(F)c1 N1(C(CCOC)=O)CCCC2(C1)CN(C(=O)CCc1ncccn1)CCO2 C1(CCC)CN(C(C2C(NC(C3C4(CC4)C34CC4)=O)C2(C)C)=O)CCO1 CS(=O)(=O)CC(=O)N1CC(O)(CNC(=O)C(O)Cc2cnc[nH]2)C1 CCC(CC)(CC)C(=O)NCCCCC(=O)N(C)Cc1sccc1C N1(C(CC(C(=C)C)OCC)=O)CCC2CN(C(c3ccoc3Cl)=O)C2C1 CC(CC(=O)NC1(C2CN(C(=O)CC3(C)CCOCC3)C2)CC1)C(C)(C)C N1(C(c2c(C)sc(C)c2C)=O)CCN(C(=O)C(C)C#N)CC(O)C1 O=C1COC(CNC(C2CC(O)CN2C(=O)CCc2ccccn2)=O)CN1 CC1(C(=O)NCc2c[nH]nc2C(=O)NCC2CC2(Cl)Cl)SCCCS1 c1(OC)ccc(OC)c(CCC(=O)NC2CC2CNC(c2c[nH]c(C#N)c2)=O)c1 Cc1cc(C#N)cnc1C(=O)NCC=CC(=O)NCc1ncc(Cl)cn1 C(=O)(CC(C)(C)C#N)NCCCN(C1CCCC1)C(C1(CC#C)CCCC1)=O C(C)(C)(CCC(=O)NOCC(F)(F)F)NC(CC(C(C)=O)(C)C)=O N1(C(c2cc(C(F)F)cs2)=O)CCCCC1c1ccc(CO)o1 c1(CN(c2nc(C)cc(OCC)n2)CC2(C)CNC2)ccc([N+](=O)[O-])c(C)c1 c1(C(=O)NC(CC)CNC(=O)CN2C(C)CCCC2C)ccc2nnc(O)n2c1 N1(C(CC=C(C)C)=O)CCOC(C(N2CC3(CCC3O)C2)=O)CC1 c1(C(NOCC(C)(C)O)=O)ccc(CNC(C2C3COCC23)=O)cc1 N1(C(c2c(OC)cnnc2)=O)C2CCC1CC(C(=O)NCC1(F)CCOC1)C2 C(CCCCC(=O)N1CC(NC(c2c[nH]c(=S)cn2)=O)CC1C)OC c1(CC(=O)NC2CC(CNC(CCCC(=O)NC)=O)C2)ccc2c(c1)OCO2.NCO c1(C(=O)NC2C=CC(CNC(C(C=C)(C)O)=O)C2)cc(C)n(CC(F)(F)F)c1C CC1(NC(C2CCN(C(N)=O)C2)=O)CCCN(C(c2cccc(F)c2N)=O)C1 N1(C(C(CCC)OC)=O)CCN(C(c2[nH]ccc2-c2ccccc2)=O)CC1C N1(C(c2nn(C)c(Cl)c2C(F)(F)F)=O)CC2CC(C1)N(C(=O)C(C)(C)O)C2 C(=O)(CC(O)CCC(C)CC)NCC1(O)CN(C(CC2(OCC)CC2)=O)C1 C1(C(=O)NC2CC(F)(CNC(CS(CC)=O)=O)C2)CC(F)(F)C1(C)C C=CCCCCC(=O)NCC(CO)NC(c1cc(OCCOC)ccc1N)=O c1(C(=O)NC2C3CN(C(C4SCCS4)=O)CC23)cc2c(s1)CCC2 N1(C(C(C)CF)=O)CCN(C(c2ccccc2Cn2cccn2)=O)CC1CCO C(CC(C)(C)C(=O)N(C(C)CNC(=O)C(C)(C)c1ccccn1)C)SC S(=O)(=O)(c1c[nH]c(C(N2CCCC(NC(=O)C(C)(C)C)C2C)=O)c1)NCCOC c1(CNC(c2[nH]ccc2N(S(=O)(=O)Cc2ccccc2)CCO)=O)sc(Cl)nc1Cl C(=O)(C(C)CC(C)(C)C)NC1C2CN(c3c(CC)c(Cl)ncn3)CC21 c1(CSC2(NC(=O)NCC3C(SC)C3)CC2)cccc(C(=O)NCF)c1 C=CC1CCCN(C(=O)C(C2CCN(C(=O)C(C)(C)CCC)C2)C)C1 c1(C(=O)NCC2CN(C(CCCN(C)C)=O)CC2(C)C)ccc2nc[nH]c2c1F C1(NC(CN(C(C=CC)=O)C2CCC2)=O)CN(C)CC1O C1(C(=O)NCCOCCOCCOCCOCC=C)CCC(=O)NC1 Cc1nnc2n1CC(C(=O)NC1(CCNC(C3(CO)CC3(F)F)=O)CCC1)CC2 c1(CC)nc(C)oc1C(=O)N(C(CC)CC(=O)NC(C)(CC)C(N)=O)C C1(C(=O)NCC(=O)NC23CCC(CC2)C3)CCOC(=O)CC1 c1(NC(C2C(C(C)NC(CS(CC)=O)=O)C2)=O)c(CO)cccc1F C1(NC(CC2ON=C(CC)C2)=O)CCCN(C(C2(C)CCC(=O)N2)=O)CC1 C1(CCNC(c2sccc2C(F)F)=O)CCCN(C(C2CC2F)=O)C1 C1(C)(NC(Cc2c(C)nn(C)c2)=O)CCCN(C(c2ccoc2C(C)C)=O)C1 C(=O)(C1CSc2ccccc21)NCCCN(c1cc(C2CC2)ncn1)C(C)C C1(CNC(=O)C(F)F)CN(C(c2sccc2-n2cnnn2)=O)CC12CC2 c1(C(=O)NCC(=O)NC2C(C(C)(C)C)=NO2)cnc(O)n(C2CC2)c1=O CCC(N=c1nc2c(cnn2C)c(NCC2CC(=O)N(C)C2)[nH]1)C1CCCC1 Cc1oc(Cl)nc1C(=O)NC1(CNC(C2CCCNC2=O)=O)CCOC1 N1(C(C2=C(C)CC2)=O)CC(CNC(c2conc2C(C)(C)C)=O)CC(C)(C)C1 C(=O)(C(CNC(c1csc(O)n1)=O)C(C)(C)C)NCC(C#C)CC c1(C(=O)NC2CN(C(=O)Nc3ccc(C)cc3)CC(F)C2)ccc2scnc2c1 NC(=O)C1=NOC(CNC(=O)NCc2ccc(Cl)cc2O)C1 c1(C(=O)NC2C(C)CCN(Cc3cccc(CC)c3)C2)cccc2nccn12 CC1(C)CCCCCC1NC(=O)C(c1ccccc1)NC(C1(C)CCCCC1)=O CC1CN(C(c2n[nH]cc2Cl)=O)CC(C)CN1C(c1ccc(F)c(C2CC2)c1)=O c1(C(C)C)ccc(CCC(N2CCC(NC(C3CNC(=O)C3)=O)C2)=O)cc1 N1(C(c2c(OC)cc(C)cc2)=O)CC2CCCC1C2CNC(C1CC1(C)Br)=O C(=O)(C(O)CCNC(=O)N(C1(c2ccncc2F)CCC1)C1CC1)OC Cc1ccc(Cn2nc(-c3cncs3)nc2Cn2ncc(Br)n2)cc1 c1(CC(=O)NC2CCN(C(CCC#C)=O)CC2F)nn(C)c2ccccc12 N1(C(C(C)C(C)S(C)(=O)=O)=O)CC(NC(=O)CCCC(N)=O)Cc2ccccc21 N(C(=NCCC1CCOCC1)NC1CCCC(C)(C)C1)CCCOC N(C1COc2ccc(Cl)cc21)C(C)CCN(c1cc(C2CC2)ncn1)C CCC(C(=O)NC12CN(C1)CC2)N1CCCC1=O.C(C)(C(C)C)=CC(=O)NC CCCCC(F)C(=O)NCC1CCCCC1NC(c1cnc(C(C)(C)CF)o1)=O c1(OCC)cc(N2CCCCC2CNC(=O)C=C(Cl)Cl)ncn1 c1(C(=O)Nc2cccc(CNC(C3(C4CC4)CCC3)=O)c2)cccc2oncc12 C(=O)(C(C)CC(C)(C)C)NCC#CC(=O)NC1C(C)NC(=O)CC1 C1(NC(c2ccc(SC(C)C)cc2)=O)CCC12CN(C(c1nocc1Cl)=O)C2 CC1(O)CCCN(C(C2CN(C(C34C=CC(CC3)C4)=O)CCN2C)=O)C1 C1(NC(=O)OCC)CC12CC(C(=O)NCC(F)CNC(=O)CC1CCC1)C2 Cc1cc(Cl)c(C(=O)NC2CCCC(CNC(c3ccn(C)n3)=O)C2)cc1C c1(C2(C(=O)NCCC(C)NC(=O)CC34CCCC3C4)CC2)ccccc1F CCCC(F)C(=O)NC1CN(C(=O)CC2CC(C)C2)CC1CCC C1(C(C)(C)C)CCC(C(=O)NC2(C3CCCN3C(C3CC3F)=O)CC2)O1 C1(CS(=O)(=O)NC)CCC(C)N(C(=O)CCCO)C1.C(C)(C)(C)OC=O c1(C(N2CCCC(NC(=O)Cc3cncnc3)C2)=O)cccc(F)c1Cl C(=O)(CC(C)(C)COC)N1C(CC)C(C(=O)NCCc2cccc(F)c2)CC1 N1(C(C2CCN(C(N)=O)CC2)=O)CCC(NC(=O)C=CI)C(F)C1 CC(C)(C)[Si](C)(OCC(=O)N=c1nc[nH]s1)c1cccc(Br)c1 C1(C(N(CCC(=O)NCC2CC2)C)=O)CCCC12CCC2.C(CCC(=O)OC)NC=O c1(C(=O)NC2CC(NC(C(CCC)CC3CCCC3)=O)C2)n[nH]c2cccnc12 c1(C(N2CCC(CCC(=O)NCCC(C=C)C)C2)=O)cc(C)n(C)c1C CCC(C)(O)C(=O)NCC1CCN(C(C2(C(=O)N(C)C(C)C)CC2)=O)C1 C=Cc1ccc(C(=O)NCC(C)NC(c2cnc3n2CCC3)=O)cc1 C(CN=c1cccc(S(=O)(=O)N2CCCC2)[nH]1)Oc1ccc([N+](=O)[O-])cc1 C1(CNC(=O)CCc2cnn[nH]2)C=CCN1C(C1(c2ccccc2)CCOC1)=O C(C(=O)N1CCCc2nccn21)SC1CN(C(C2(C)CCCC2O)=O)C1 C(=O)(CC(C)OC)NCC(c1ccccc1)CNC(C(F)=CC)=O CC(CS(C)(=O)=O)C(=O)N(C1CN(C(c2cnc([N+](=O)[O-])n2C)=O)CC1(C)C)C c1(CSCC#N)cc[nH]c1C(=O)OCCOC(COC)=O C1(C(=O)NC(C#CCC)(C)C)CC(NC(c2cc[nH]n2)=O)C12CCC2 C1(C)(CNC(C=CC(C)C)=O)CC(NC(c2cc(-c3cccs3)on2)=O)C1 N1(C(C=CCN(C)CC)=O)CCC2(CC1)CC2NC(c1ccc(N(C)C)cc1)=O CC(C)(CNC(=O)CC1COC(=O)C1)CC(=O)NC(c1ccccn1)CO N1(C(C2(C)CCCC2O)=O)CCCN(C(c2ncc(F)cc2F)=O)CC1 N1(C(C(CC(C)C)(C)C)=O)CCC2C(CCN2C(c2ccc(F)n2C)=O)C1 CC(C)CC(C)C(=O)N1CCSCC1C(=O)NCC(C1CCCC1)O CC(c1cccnc1)=CC(=O)NC1CCCC1NC(=O)CCNC(=O)CO C1(CC)C(NC(c2cncc(F)c2)=O)CCCN1C(c1ncn(C)n1)=O C1(C(=O)NC(CCNC(c2scc(C(=O)OC)c2)=O)C)CCC(C(C)(C)O)CC1 C(=O)(C(O)C(F)(F)F)N(CCC(C)NC(c1cc(CN(C)C)on1)=O)C C1(CC(=O)NC(CC(=O)NC(c2nc(=O)o[nH]2)C)C2CC2)CCN(C)C1=O C(=O)(C(O)CC(C)C)N1CC2C(COC(C3(CCOCC)CCC3)=O)(C2)C1 CC1CCCC(CC(=O)NCc2cn(Cc3nc(C(=O)O)cs3)nn2)C1 c1(CCC(=O)NC2C=CCN(C(C3C(C)(C)OCC3)=O)C2)cc2ccccc2o1 CCC(C)CC(C(=O)N1CC(c2nn[nH]n2)C1)NC(c1csc(=N)[nH]1)=O N1(C(CCOCC)=O)CCC2CCN(C(c3cc(C(C)C)nc(O)c3)=O)CC2C1 N1(C(c2cn(CC)nn2)=O)CCC(NC(c2cc3c([nH]2)CCC3)=O)C2(CCC2)C1 c1(C(=O)NC2CN(C(C3CCCOC3)=O)C2)cc(Cl)c(Cl)[nH]1 C1(CC(=O)N(C2CCN(C(c3nc(=O)n(C)[nH]3)=O)C2)CCC)C=NN(C)C1=O C(=O)(C1=C(Cl)CCOC1)N1CCN(C(c2c(C)nn(CCO)c2)=O)C2C1C2 Cc1cccc2c1CN(C(=O)C(F)CC1CN(C(=O)CC3OCCC3(C)C)C1)C2 c1(C(=O)NCC2(NC(CC=C)=O)CCCCC2C)cnc2n(c1=O)CCS2 C12CN(CC(C)(C)O1)C2=O.c1(CN2C(COC)CCC2)ccc(C(N)=O)cc1 c1(OC)cccc(C(=O)NC(C2CN(C(=O)CC#N)C2)C)c1OC C(=O)(CC(C)C(F)(F)F)N(C1CCN(C(=O)CNS(C)(=O)=O)CC1)CCOC C=CCC(CCCCC)C(=O)NCC(C)NC(c1ncoc1C1CCC1)=O c1(C(N2CC(N(C(c3c(C)noc3)=O)C)C(F)C2)=O)cnn2cccc2c1 N1(C(C(C)OC)=O)CC2CCC1CN(C(=O)CSCC(F)F)C2 c1(N(C(CC)C)C(c2nc(C)n(C)c2C)=O)ccc2c(c1)OCO2 C1(NC(C(C)N(C)C)=O)CN(C(=O)Cc2nnn(C(C)(C)C)n2)CC1C CC(CNC(=O)C(C1(O)CCCC1)F)C(=O)N(C)CCN(C)C1CC1 O=C1CCC2(CN1)CN(C(=O)COCCNC(C1CC3(CCC3)C1)=O)C2 C1(C#N)(C(N2CCC(CN(C(=O)COc3ccn(C)n3)C)C2)=O)CCCC(=O)C1 C1(C(N(CC)CC)=O)C(Cl)(Cl)C12CC2.C(C)(CN(C(=O)CN)C)NC(=O)C1CC1 C1(OC)CC(CCNC(c2c(C)coc2C)=O)N(C(c2ccc(SC)cc2)=O)C1 c1(C(=O)NC2C(C)CN(C(c3cnc(Cl)s3)=O)C2)n[nH]c2c1CCC2 N1(C(CCC)=O)CC(C(=O)Nc2cc(C(C)C)ccc2O)CC(F)C1 CC1C2C(CCN2C(=O)CC#N)CN1C(=O)C#CC1CCOC1 N1(C(c2c(C)[nH]nc2CO)=O)CCC2(COC(CNC(=O)C3=NOCC3)C2)C1 c1(OC)cc(-n2nc(CC3CC3)nc2C2CC23CCOCC3)cc(Br)c1 C(C(C)(C)C(F)(F)F)NC(c1nnnn1Cc1ccccc1)C1(SC)CCC1 C1(C(C)C)CN(C(=O)Cn2ccnc2)CC1C(=O)NC(C)Cc1cn[nH]c1 N1(C(C2C(C)C2)=O)CCN(C(C2(c3cn(C)nn3)CC2)=O)C2COCC12 C1(NC(c2n(CC)ccc2)=O)CCC(O)CN(C(=O)CCCCOC)C1 c1(CNc2nc(N(C)CC)nc(N3CCCC(C)CC3)c2)cccc2c1OCO2 C1(C(=O)Nc2cc(C)cc(C)c2)N(C(C2CCC3(CCC3)C2)=O)CC12CCCC2 C1(C(=O)NCC(CNC(CSCC)=O)F)COCC1n1ccnc1 C(CNC(C1(Cl)C2CCC(=O)C12)=O)(CC(F)(F)F)NC(c1csc(O)n1)=O C1(C(=O)NC2CC(CCNC(C(CCCC)O)=O)C2)CCc2nnc(C)n2C1 c1(C(N2CCC(C)(NC(c3cccc(N)n3)=O)C2)=O)ccc2cccnc2n1 Cc1cc(NC(C2CCC3(CC3)N2C(=O)C=Cc2cc[nH]n2)=O)ccc1O Cc1nc2c(C(=O)NCCC(C(C)C)NC(=O)C=CI)ccnc2[nH]1 c1(CN(C(CC=C=C)=O)C23CC(c4ccc(F)cc4)(C2)C3)nc(Cl)c(CSC)[nH]1 C(=O)(CC(C)(C)C(C)(F)F)NC(C)CN(C(=O)C(C)Oc1cccc(F)c1)C c1(OC)cccnc1CN1CCC(n2nnnc2C(C(C)C)OC)CC1.C(F)(F)F Cc1cccnc1CC(=O)NC1CCC(NC(=O)CC2CCCC23CC3)CC1 c1(C(C(=O)NCCCC)N(C(CC)C2CC2)C)cccc(CSC)c1 C1(C(N(CCNC(C)=O)C)=O)(N(C(=O)CSC(F)F)C)CCC1 c1(C(=O)NC2CN(C(CC3(C=C)CCC3)=O)CC2CC)cnc(C(C)C)nc1C N1(C(=O)NCc2cccc(OC(C)C)c2)CCc2ccc(CC)cc2C1 CC1CCC(C(N2CCC(C(F)F)CC2)=O)CN1C(c1cnnc(O)c1)=O c1(NC(C2N(Cc3cccc(C)c3)CC2)=O)ccc2c(c1)OCCN2C c1(NC(c2ccccn2)C(=O)N(CCCCN(C)C)C)ccnc(C(=O)O)c1 C1(C(=O)NC(CC)Cc2cccc(Cl)c2)CCN(C(=O)OC(C)(C)C)C1(C)C c1(CN2CCC(CNC(=O)C(c3ccc(F)c(F)c3)O)C2)c(F)cccc1F c1(N(CCOCC)C)nc(N2CCOC(C(C)C)CC2)nc2sccc12 c1(C2(C(=O)NCCN(CCC)C(C3CCC(=O)O3)=O)CCC2)ccc(F)cc1F O=C1COc2cc(C(=O)NCc3cccn4c(Br)cnc34)cnc2N1 CCC(CCOC)C(=O)N1CCN(C(=O)C=CCOC(C)(C)C)C(C2CC2)C1 N1(C(c2cc(C(N)=O)ncc2)=O)CC2(CNC(C3(C(F)F)CC3)=O)CCC1CC2 N1(C(Cn2c(C)cc(C)n2)=O)CC(CC(=O)NCC(C)(O)C(F)(F)F)CC1(C)C c1(C(=O)NCC2C3CCC(C3)N2C(c2ccoc2Cl)=O)cc2c(nn1)CCCO2 N1(C(C2N(C(C(CCC)NC(N)=O)=O)CC(C)C2)=O)CC(O)CC(O)C1 C(=O)(CS(=O)(=O)Cc1ccc(Cl)s1)NC(C)CN(C)C(c1cnsn1)=O N1(C(=O)CCc2ccc(F)nc2)CC2(CCCCN2C(=O)CC2CCC3CC23)C1 Cc1cc(CCC(=O)NCC(C2CCOC2)NC(=O)C(C)(C)n2ccnn2)n[nH]1 C1(CC(=O)NC2C(N(C)C)CCC2)C2CCC(C2)N1C(c1cc(C2CC2)on1)=O C1(CCCC)CN(C(c2cnn(CC)c2)=O)CCN1C(=O)C(C)CC(=O)OCC C(CNC(=O)CC1(C)CCOC1)(CC(=O)N(C)CCOC(F)F)OC Cn1ncc2c(N(C3CNCC(F)(F)C3)C(c3ncon3)=O)ncnc12 c1(CNC(C2C(NC(C3CN(C(C)C)C3)=O)C2)=O)c[nH]c2cccc(Br)c12 C1(NC(C(c2ccccn2)C)=O)CC(C)N(C(=O)CCCc2csc(=N)[nH]2)C1 c1(-c2onc(N(C)C)n2)cccc(S(=O)(=O)N2CCCCC2C2(O)COC2)c1 n1(CCNC(CC2N(C(=O)NC3CC(OC)C3)CC2)=O)cc(Br)cn1 n1(CC)cc(Br)c(C(=O)N(CC(C)NC(=O)C(C(C)C)n2cnnc2)C)n1 C(=O)(C(C)(C)CC1CCC1)N1CCC(CCCNC(=O)COCC2CCOC2)C1 Nc1ccc(C(F)(F)F)nc1C(=O)NCCN(C(=O)Cc1ccncc1)C1CC1 c1(C(=O)NCCCN(C)C(C2C=CC=CC=C2)=O)cc2c(nc3ccccn23)s1 CCCCC(CC)CC(CC)NCc1cnn(C2CCOCC2)c1C C(=O)(CCCC(C)=O)NCCN(C(=O)Cc1cccc(OC)c1)CCC n1(CC)ncc(NC(N(C)C(=O)OC2(CO)CCOC2)=O)n1 c1(NCC2COCN(C(C)C)C2=O)[nH]c(=NC2COCC2C2CC2)nc2sccc12 CC1CC(NC(c2ncc(C(F)(F)F)s2)=O)CN1C(c1ccnnc1Cl)=O c1(C(=O)NC2CCC(CCNC(C=CCC)=O)C2)ccc(NS(C)(=O)=O)nc1 C(=O)(C1=CCC(C)(C)CC1)N1CC(C(=O)NCC(CC(=O)NC)C)OCC1 c1(C(N2CC(C(=O)Nc3ncc(C)cc3C)C2)=O)cc(Cl)nc(Cl)c1F N1(C(C(CCC)C(C)C)=O)CCCC12CCN(C(=O)C1CCc3scnc31)CC2 C1(NC(c2cnc(CC(C)C)[nH]2)=O)CN(C(=O)Cc2ccnnc2O)CC12CC2 N1(C(c2c(NC)cnnc2)=O)CCC(C(=O)NCCC(C(C)C)OC)CCC1C Cc1ccc(N2CCCC2)c(C23CC(N(C(=O)CCCS(C)(=O)=O)CC)(C2)C3)c1 C12(NC(C3C(COC)C3)=O)CCC(CNC(=O)CN(C)C(C)=O)(C1)OC2 c1(COC(C(N2CCCNCC2)C)=O)cnn2c(Cl)cccc12 n1(CC(=C)C)nc(Cc2ccc(C)cc2)nc1-c1cn(CCO)cc1C C(=O)(C(CC(F)(F)F)c1ccc(F)cc1)NCCN(C(=O)CP(C)(C)=O)CCC c1(NCC(CCCC)NC(=O)Cc2c(Cl)cnn2C)ccc(C(=O)OC)c(C)c1 C=CCC(CC)C(=O)N1CC(NC(=O)CC23CCC(CC2)CC3)CC1C c1(C(N(C)CC2CN(C(C3CC=CCC3)=O)CCO2)=O)cnc2occc2c1 C1(C(=O)NC(C2(C(N3CCC(N=[N+]=[N-])C3)=O)CC2)C)CCC2(CCC2)O1 CC1CCN(C(c2cnn3ncccc23)=O)CCN1C(=O)CCc1cn(C)cn1 C(=O)(N=c1[nH][nH]c(C)c1C)c1c(C(N=c2[nH]ncc(C)c2)=O)nccc1 c1(OCC)ccc(C(=O)NC2CC(NC(C)=O)CC2O)cc1S(N)(=O)=O N1(C(C2(C(=O)NC)CC2)=O)CCC2(CCCN2C(=O)Cc2cccc(C)c2Cl)C1 N1(C(COCCC=C)=O)CCC(C(C)NC(C2C=CCS2)=O)CC1 c1(C(=O)NC2C(C)CN(C(c3ccc(Cl)cn3)=O)C2)cc2ncccn2n1 c1(C(N2CCC(NC(=O)COC3CC3)C2)=O)cccc(C#CC2CC2)c1 CCCC(CC)C(=O)N1CC(C(=O)Nc2ccc(OC)cc2C)C(F)(F)C1 C1(NC(c2cc(CC)no2)=O)CCN(C(C2CCC(C(N)=O)C2)=O)CC1CO C(=O)(CC(CN(C)C)CC)NCC(CC)NC(=O)CN1CCSCC1 C1(NC(C(C)OC)=O)CCN(C(C2CCCN2C)=O)C1C CC(CO)C(=O)NCC(C1CCC1)NC(=O)CSCCCc1ccccc1 Cc1ccc(NC(C2CC=CCN2C(C2CCC2C#N)=O)=O)c(C)c1 C1(C(=O)NCCOCCC(C)C)CCN(C(C2CCCS2)=O)C1 C(CN=c1[nH]c(NC2CCCC2S(C)(=O)=O)nc2ccsc12)N(CCCC)C C(=O)(CC1OCCc2ccsc21)NCCOCCN(C(C(C)(CO)OC)=O)C c1(CCC(=O)NCC2CN(C(=O)C3=C(Cl)CC3)C2)n[nH]c2c1CCCC2 c1(CNC(C(c2ccccc2F)OC)=O)ccccc1CNC(=O)CCSC N1(C(C(CC)Oc2ccccc2)=O)CCC2(CC1)CN(C(=O)CSC(C)C)C2 n1(CC)cc(C(=O)NCCOC(C)(C)CNC(=O)CC2C(=O)NN=C2C)c(C)n1 CC(CC(C)(F)F)C(=O)NC1(C2CN(C(C3COC(C)(C)CO3)=O)C2)CC1 c1(NC(C2N(Cc3[nH]c(C)c(C(=O)O)c3C)CCSC2)=O)ccnc([N+](=O)[O-])c1 Cc1cc(Cl)ncc1CC(N1CCCC1c1cn(Cc2ccc(F)cc2)nn1)=O C(=O)(C(C(C)C)c1noc(C2CC2CC)n1)NC(C1(C)OCCO1)CC c1(C(N(C2CCN(C(c3cc4c(s3)CCOC4)=O)C2)C)=O)nc2ccccc2[nH]1 C1(NC(C(CC=C)CC)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)CC1(C)C N(C1CN(C(c2c(F)c(C)nn2C)=O)CCc2ccccc21)C(CCOC)=O c1(C2C(CNC(CC3(CNC(COCCC)=O)CC3)=O)C2)ccsc1 c1(OC)c(F)c(C(N2CCC(NC(C3C4COCC34)=O)C23CC3)=O)cc(F)c1F N1(C(c2cn(C3CC3)nn2)C(=O)CSC)CCC(O)C1C.C(=O)(OCC)NCC n1(CC=C)cc(C(=O)NCC(C)(C)NC(=O)C(F)OC(F)(F)F)cn1 c1(CC(=O)NCCOc2ccc(Cl)c(Cl)c2)c[nH]c2c(Br)cccc2c1=O c1(C(N2C3(CN(C(c4cc(C)ncc4)=O)C3)CC2)=O)cc(C)cc(Br)c1N c1(C(=O)NC2C(CO)CCN(C(c3n[nH]c(C)c3C)=O)C2)cnc2ccoc2c1 C(C(C(C)(C)C)NC(=O)CCc1cccs1)NC(COCCCC)=O C1(C(=O)NC)CCCCC12CCC2.c12cn(nn1)C1CC23CC13.C(=O)(NC)NC C#Cc1cc(F)c(C(N2CC(NC(C3(C)CC(F)C3)=O)C(C)C2)=O)c(F)c1 c1(C)cn(CC2CN(C(CC3C(OC)CC3)=O)C2)nn1.c1(S)nc(C(=O)O)cs1 Cc1c(-c2ccc(C3(C(N4CCC5(CCC5)C4)=O)CC3)cc2)cc(F)cc1F c1(OCC)cnc(OC)nc1.c12ccnc(n1)C(=O)N2C1CNCC(C)C1 C1(NC(C(COC)O)=O)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1(C)C C(C)(C)(CC(=O)N(CCNC(C1C(C)C1(F)F)=O)Cc1ccccc1)OC Cn1c(NC(C2CCc3cccc(Br)c3C2)=O)cc2ccccc12 C(=O)(C1=C(Cl)CCC1)NC1CN(C(CCC2CC(OC)C2)=O)CC1C c1(C(=O)NCC(C)(C(C)C)NC(CC(CCC)C)=O)noc2ccc(Cl)cc12 Fc1ccc(CNCC23CCCCC2C3)cc1C(F)(F)F CC1CN(C(C2OCCC2NC(C2CC2(F)F)=O)=O)CC(C)(C)O1 C1(F)(CNC(c2ccnn2CCF)=O)CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC1 c1(OC)nc(C(=O)NCC2CC(NC(c3cnoc3C)=O)C2(C)C)ncc1F CC1(C)CCC(C(=O)NCCOC2CCN(C(c3cc[n+]([O-])cc3)=O)C2)O1 c1(CC(=O)NC(CC(C)C)CNC(=O)C(C)N(C)C)cccc(Cl)c1Cl C1(O)(CNC(C2C=CC(NC(C(C=C)O)=O)C2)=O)CC2CCC1C2 c1(OCC#C)ncccc1C(=O)NCC(C(C)C)NC(C1CC1C(F)(F)F)=O Cc1ncccc1C1C(CO)C1(C)C.C12CCN(C(=O)OC(C)(C)C)C1NC2 N1(C(C(C)N(C(=O)C(COC)NC(C)=O)CCC)=O)CC2CSCC(C2)C1 c1(C(=O)NCCNC(c2ccc(C(C)(C)C)[nH]2)=O)cnc(O)c(Br)c1 c1(C(N(CC(CNC(C(C)NC(COC)=O)=O)O)C)=O)cnc(N)cn1 C1(CNC(c2c[nH]nc2[N+](=O)[O-])=O)C(O)C(O)CN1C(=O)COCC1CCCO1 CC1CN(CC(=O)Nc2ncc(-c3ccc(C(F)(F)F)nc3)cn2)CC(C)O1 C(C(C)N=c1[nH]nc(C(C)(C)C)o1)N(CC)Cc1ccccc1 C(=O)(CCCCC(=O)N1CSCC1C(=O)NC(CN(C)C)CCO)OC c1(OC)ccc2c(c1)C(NCc1cn(C)cn1)CCCO2 c1(OC(C)C(=O)N(CCCN(C)C(c2ncccc2F)=O)C)ccc(F)cc1Cl C1(NC(CC2(C=C)CN(C(C3CSC(C)C3)=O)C2)=O)CCC2(CCC2)C1 Cc1cccc(C(C)CNC(N2CCCC(O)C2)=O)c1 CC1CN(C(c2cc(Cl)ccc2Cl)=O)CCC1N(C(=O)CCCF)C N1(C2CC3(CC(O)(C(F)(F)F)C3)C2)CCn2c(cnc2-c2ccccc2)C1 c1(C(=O)NC(CNC(C2(O)CCOCC2)=O)CO)nc(Br)sc1Cl C1(N(C(=O)CSC)CCOC)CCN(C(=O)CC(C)c2ccccc2)C1 C1(CN2CCN(C(C3C4CN(C)CC43)=O)CC2)OC(=O)CC1(C)C Cc1ccc(F)cc1C(=O)NCCC1CN(C(C2CCC(=O)N2)=O)CC1C N1(C(CN(C2CCSCC2)C)=O)CCCC(O)(C(=O)NCCc2ccncc2)C1 C1(C(=O)Nc2cscc2C2N(C(CSCC)=O)CC(OC)C2)CC2C(C1)C2(F)F C1(CC(=O)Nc2nccn2C)CCN(C)C1.C12(CCC1)CNC(=O)CN(C)C2 Cc1cc(N2CCC(Cc3nccc(O)n3)C2)nc(=NCC2CNC(=O)C2)[nH]1 Cc1ccc(C(=O)NCCC2CN(C(=O)Cn3cc(C4CC4)cn3)CCO2)nc1 c1(C(=O)NC(C(=O)N(C)Cc2ccc[nH]2)C2CCCC2)cn(CCO)nn1 N1(C(c2cn(C)nn2)=O)CCCC(CO)(NC(=O)C2=NOC(c3ccccc3)C2)C1 c1(C(=O)OC)cc2c(N3CCC(CCNC(c4ccoc4)=O)C3)[nH]cnc-2n1 C1(C(N(C)Cc2cccc(-c3nn[nH]n3)c2)=O)CCCC(C)(C)CC1 N1(Cc2cn(Cc3c(OCC)c(CO)ccc3C)nn2)CCCC2(CCCO2)C1 c1(C(=O)NC(CCNC(C2(OC)CCCCC2)=O)C)cccc(C(C)C)c1F c1(CN2CC3C(NC(c4c(N(C)C)cccn4)=O)C3C2)ccc(O)c(F)c1F C1(C(=O)NC2CCCN(C(C=Cc3nc(C)sc3)=O)C2)CCC(C)(C)CC1 C(CCC(=O)NC(CC1CN(C(=O)OC)C1)C)NC(=O)C(F)(F)c1cscn1 C1(C(N2CC(C)SCC2)=O)CC(F)CCN1C(=O)CN1CCC(O)CC1 N1(C(C2CC(C#N)C2)=O)CCC2(CCCC2NC(c2ccon2)=O)CC1 c1(NC(c2cc(C)c(Cl)c(N)c2)=O)ncnc2sc(Br)cc12 N1(c2nc(SC)nc(Cl)c2)CC(CNC(=O)CC2CCC(=O)N2)OC2(CCC2)C1 CN1C(=O)COCC1CNC(C1CC2(CC2)CN1C(=O)CC1CC2(CCC2)C1)=O c1(C(N(C(C)CNC(=O)CN2CC3CCC2C3)C)=O)ccc2cc(F)ccc2n1 N1(C(Cc2ccc(OC)c(O)c2)=O)CCCN(C(=O)C2=NOC(C)C2)C(C)C1 CC1(C)COC(CCC(N2CCCC(NC(=O)CCc3cc(Cl)no3)C2)=O)C1 N1(C(c2c(CC)onc2)=O)CCCC(CO)(NC(c2ncc(N)cc2C)=O)C1 CN1CCc2c(C(=O)NC3CCN(Cc4cccc(C#N)n4)C3)cccc21 CC(C)CS(=O)(=O)CCC(=O)N1CCCC(N(C(=O)CSCCC#N)C)C1 C1(CO)C2CCCC2CN1C(=O)CC(C)(C)C(F)F.c12cn(nn1)C2C c1(C(N2CC(C(C)NC(c3cccnn3)=O)C2)=O)ccc(Cl)c(Br)c1 c1(OCC(=O)NC(C)(CNC(C23CC(O)C2C3)=O)C2CC2)c(F)cccc1F C(=O)(CC1COc2ccccc21)NC(C)CCNC(c1c[nH]nc1F)=O C1(CNC(C(COC)C)=O)CCCCN(C(=O)CCc2cc(C)cc(C)c2)CC1 CC(CCC(=O)NC1CC=CC1)NC(=O)C(F)C1CCCC1 C1(CCOC)CN(C(=O)Cc2c[nH]nc2C)CCN1C(=O)CSc1cn[nH]c1 c1(C(=O)NCC(C2(O)CCN(C(C3(CO)COC3)=O)C2)C)cncc(C2CC2)c1 CN1C(=O)CCCC1C(=O)Nc1cccc(CC(=O)NCC2CC2)c1 c1(CN2CC(OC)C(NCc3ccc(C(=O)O)o3)CC2)cc2ccc(Cl)cc2[nH]1 C1(F)(CNC(c2cccc(Cl)c2)=O)CCCN(C(C2CCOC2C2CC2)=O)C1 c1(OC)cc(F)c(C(=O)NC2CC(F)(CNC(=O)C=Cc3cccs3)C2)cc1OC C(CCC(C)C)(C(=O)N1CC2CC(NCc3ccc(C4CC4)o3)C1C2)NC(C)=O C1(CNC(=O)C2=CCCCC2)CC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)CO1 C=CCC(C)(CC)C(=O)NC1CC(C(C)NC(=O)CCC(CF)CF)C1 C1(C(=O)NC)C2C3CC4C1C2C34C(=O)NCc1ccc(Br)nc1.C1CCN1 CC(C)CC(C)C(=O)N1CCCC1CCC1CCCCN1C(c1cccs1)=O c1(C(=O)NCC2N(C(C(CC)F)=O)CCC2)cnc(SCc2ccccc2)[nH]c1=N N1(C(CCCCC)=O)CC(C(=O)NCCCN(C)C(C)=O)CCC1C C(=O)(CC(O)C(C)C)N1CCN(C2CCN(C(CNC(CCOC)=O)=O)C2)CC1 c1(C(CNC(c2cc(C)c(Cl)s2)c2nnnn2CCCF)C)ccc(Cl)c(Cl)c1 N1(C(C=CNN(c2ccc(C)cc2)C2COCCO2)=O)CC2CNC2C1.C(C)=O N1(C(COc2ccc(NC(C)=O)cc2)=O)CCC(C)C(NC(=O)CC#N)C1 C1(NC(=O)CN2CCC2)COC2(CNC(=O)C(O)c3ccco3)CC1C2 CCC(CC(=O)N1CCC(C(=O)NCc2nncn2CCO)(CC)C1)C(F)F c1(NC(C(c2ccccc2)NC(C2(COC)CC2)=O)=O)cc(C#N)c(Br)cn1 c1(OC)cccc(C(N2CC=CC(NC(=O)C(C)CSC(F)(F)F)C2)=O)n1 C#Cc1ccc(CC(N2CC(N(C(=O)C(C)NC(C3CCCC3)=O)C)C2)=O)cc1 C12(C(=O)NC(C3CCOC3)CNC(C=Cc3cc(C)no3)=O)CC(C)(CCO1)C2 c1(OCC=C)ccccc1C(N1CCC(N(C)C(C2CNC(=O)N2)=O)CC1)=O c1(C(=O)NCC(CC(C)C)NC(c2ccc(CC)s2)=O)nn(C)c(C)c1Cl n1(CC(=O)NC(C)(CNC(=O)C=CC2CCCO2)C2CC2)cnc(C#N)n1 N1(C(c2c(C)cc(C(C)C)cc2)=O)CC2CCN(C(c3csnn3)=O)C2C1 C1(N(C(C(CC=CC)NC(=O)Cc2cnn(C)c2)=O)CC)CN2CCC1CC2 c1(C(=O)OC)cc(Cl)c(O)c(S(=O)(=O)NC2CN(C(c3ccc(F)cc3)=O)C2)c1 N1(C(C(C)n2ccnn2)=O)CC(C(=O)Nc2cncc(C(F)F)c2)CC(C)(C)C1 c1(C(N(C2CN(C(c3nc(Br)cs3)=O)CC2F)C)=O)ccncc1F CCC(=O)CCC(=O)NC(Cn1cncn1)C(=O)NCc1cccc(O)c1 c1(SCCC(=O)NC23CC(C2)N(C(=O)C2=CCOC2)C3)ccc(F)cc1 c1(CCNC(C2(C#C)CCC2)=O)ocnc1CNC(c1cnn(C(C)C)c1Cl)=O N1(C(C2(CC(C)C)COC2)=O)CC=CC(NC(=O)C2=C(C)CC2)C1 C(=O)(CCCCC#N)NC(C(=O)NC(C#C)CC1CC1)(C)C1CCC1 CCN=c1[nH]cc(C(=O)NCCCCN2CCCCC2)s1 Cc1cscc1C(=O)NC(CN(C(=O)CC1(C)CCCC1)C)Cc1ccccc1 C1(C(=O)NC23CC(NC(CC4CCC(C#N)C4)=O)(C2)C3)CCc2ncnn2C1 C(=O)(CC(C)CC(C)(C)C)N1CCCC(C(=O)NCC(CC(C)C)O)CC1 C(=O)(C(C(C)(C)C)n1cc(I)cn1)NCCCCCCSC c1(SC)cccc(NC(C2CN(C(C3(C)CC=CC3)=O)CC2C(C)C)=O)c1 c1(C(C)C(=O)NCCCN(C(=O)C=CCN2CCCC2)C2CC2)cnn(C)c1 C(=O)(C(C)(CC)C(N)=O)N(C1CCN(C(c2cc(SCC)ncc2)=O)C1)CC c1(C(=O)NCC(CNC(C23OCCC(C)(C2)C3)=O)CO)cnn2ncccc12 c1(C(=O)NC2CN(C(C=CC(CC)=CC)=O)CC2F)cnn2c1C(C)CCC2 c1(C(=O)NC(C)CNC(c2cnc(S(C)(=O)=O)s2)=O)cc(F)cc2nn(C)cc12 N1(C(C(=O)NC(C)C)=O)CCC2(CC1)CC2C(=O)Nc1cc(F)c(Cl)c(Br)c1 C1(C)(C(=O)NCC2N(C(c3cnn(C(C)C)n3)=O)CC2)CCN(C)C1 CC(C(=O)NCCC1CCCN(C(=O)CSCc2cscn2)C1)C(C)(F)F Cn1nccc(C(N2CCOC(CCNC(=O)CC3CCC34CCC4)C2)=O)c1=O CC1CN(C(C2CCS2(=O)=O)=O)CC(C)N(C(C2CCCC2(C)C)=O)C1 N1(C(C=CC(CC)C)=O)CCC(C(C)(C)NC(c2cnc(N(C)C)o2)=O)CC1 c1(C(COCCCNC(N(C)Cc2ccccc2)=O)O)ccc(O)cc1 c1(OC)cc(C(=O)N(C2CCC2)Cc2cccc(C)c2)cc([N+](=O)[O-])c1Cl C12(NC(C3C(C)C3C)=O)CCCC1N(C(=O)CC1(O)CCOC1)CCC2 C(N=c1[nH]cncc1Br)C1CN(C(C(c2cc(Cl)ccc2Cl)C)=O)C(C)C1 c1(CN(C)C(C2CC(CNC(=O)CCC3CCOC3)C2)=O)cc(Cl)no1 N1(C(c2ncn(C(C)C)c2)=O)CC(C(=O)NC(C)CC(C)(C)C)CC(C)(C)C1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)N1C2CN(C(CCS(C)=O)=O)C(CC2)C1 C1(NC(=O)C2=CCCSC2)CC2CC(C1)N(C(C13CCC(N(C)C)(CC1)C3)=O)C2 Cc1ccc(C)c(SCC(=O)NCC2CC(NC(C3COCCOC3)=O)C2)c1 C1(C(N(CC(CC)NC(CCOCC)=O)C)=O)CS(=O)(=O)CC12CC2 c1(NC(C2CC3CC3N2C(c2sc(Br)cc2Br)=O)=O)nccc2cccnc12 N1(C(COC)=O)CCCC1CN(C(=O)Cc1cnoc1)C C1(CNC(c2ccoc2Cl)=O)C2CCCC1N(C(=O)Cc1ccc(F)cc1F)C2 c1(C(N2CC(O)CC(NC(c3n(CCC)ccc3)=O)C2)=O)c(F)cc(O)cc1F CC1CC(CNC(=O)Cc2cnns2)CN1C(c1cccc(-n2cncn2)c1)=O c1(NCC(C)(C)NC(COCC#C)=O)cnc(C#N)cn1 C(=O)(C(C)C(O)C(C)C)N(CC(=O)NCC(C(C)C)OC)C c1(C(=O)NC2CCC(N(C(=O)CC3(C)CCC3)C)C2)cccc2nccn12 c1(CC)ccc(C(N2CC3CC2CC3NC(c2cc(C(F)F)cs2)=O)=O)cc1F N1(C(C=CCCC)=O)CCCC1C1CCCCN1C(c1sc(C2CC2)nc1C)=O c1(C(N(C(CNC(COCCC#C)=O)C)C)=O)cnn2cccc(Cl)c12 N1(C(C(C(C)C)NC(=O)C(=O)NC(C)C)=O)CCC2(CC1)CC(OCC(F)F)CO2 CC(C(=O)NCCC(C)NC(C1CC2(CCOCC2)C1)=O)C(F)(F)C(F)F C(CN=c1[nH]c(=NCCCF)c2cccc(F)c2[nH]1)SC(C)C C(c1ccccc1F)=CC(=O)N(C)CC1CCN(C(C2CC23CCOC3)=O)CC1 c1(C(=O)NCC2C(NC(CSc3cc(C)no3)=O)CC2)c(C)oc2ccccc12 c1(C(=O)NCC(C)N(C(c2cc(C(C)C)no2)=O)C)c2c(nn1C)CCSC2 c1(-c2c(C)noc2-c2ccn(C)n2)cc2cc(Cl)ccc2n1C c1(C(N(CC(C)NC(c2c[nH]ccc2=O)=O)CC)=O)cn2c(n1)COCC2 CCCCC(CNC(=O)C(CCC)NC(N)=O)NC(c1cc(C(N)=O)c[nH]1)=O c1(CC)nn(C)c(C(=O)NC(C)CNC(=O)CC2CC2(Cl)Cl)c1Cl c1(CC(=O)N(CC#C)Cc2nccs2)c(C=C)cc(OC)cc1OC c1(OC)cc(C(N2CCCC2C(C)(C)O)=O)ccc1O Cc1nc(C(C)C)ncc1C(N1CC2CC(NC(=O)C(C)CF)C1C2)=O c1(C(N2CCC(CN(C(=O)C(CO)N(C)C)CC)CC2)=O)c(N)cccc1F C=CC(C)(CC)C(=O)N1CCC(NC(c2cc(C3(O)COC3)on2)=O)CC1 C1(NC(=O)CCCF)CCCCC12CCN(C(=O)C(F)C(F)(F)F)CC2 Cc1cn2c(C(N3CCCCC3CNC(C3CC4C(C3)C4(F)F)=O)=O)cnc2s1 C1(CCC(=O)NCC2CCN(C(=O)CC3CCCCO3)C2)CCC(O)CC1 CC1(C)C=C(C(=O)NCC2CN(C(=O)C(c3ccc(F)cc3)F)CCO2)C1 N1(C(C(C)NC(C)=O)=O)CC2CN(C(c3c(F)cc(F)cc3F)C)CC2C1 c1(C(=O)NCC2CCCN2C(=O)Cc2nnc(O)s2)ccc(Cl)c(Cl)c1O C(=O)(CCC(CF)CF)NC12C(CN(C(Cc3nc(C)sc3C)=O)C1)CC2 c1(C(=O)NCC(CC)NC(c2n[nH]c(C)c2C)=O)ccc2ncnn2c1 C(=O)(C1=CCCSC1)NCC(CNC(CCC1OCC(C)(C)C1)=O)F C1(CC(C)C)C(=O)NC2CC(C2)C(=O)NO1.N1(C(C)=O)CCC(C(N)=O)(N(C)C)C1 c1(OC)cc(C(=O)NCC2CCC(NC(=O)CC34CCCC3C4)CC2)cc(OC)n1 c1(OC)cc2[nH]c(C(=O)OC(c3[nH]nc(CCC(=O)OC)c3Br)C)cc2s1 C=CCC(C)(C(=O)NC1CCN(C(=O)CCOc2cccnc2)CC1C)N(C)C N1(C(C2C(C)OCC2)=O)CC2(CCN(C(C3(c4ccnc(Cl)c4)CC3)=O)CC2)C1 C(C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)NC(CC(C)CC1CCC1)=O C1(NC(c2nc(C)sc2)=O)CN(C(C2CN(C3CCOC3)C2)=O)CCC12CCC2 C(=O)(C(C(=O)NC1(CCNC(c2cnc(OC)s2)=O)CCCC1)C1CC1)OCC C1(C(=O)NCCN(C(C2N(C(C)=O)CCC2)=O)C2CC2)CCn2nnnc2C1 Cc1cc(F)c(C(N2CCC(N(CCO)C(c3ccc(C#N)o3)=O)C2)=O)cc1F CC1CN(C(C2CCCN2N=O)=O)CCCN1C(=O)C=CC1CCCN1C CCCCCCC(CC)C(=O)N1CC(COC)(NC(=O)CCCCC(F)F)C1 c1(CNC(C(C(C)(C)SC)NC(=O)OC(C)(C)C)=O)ccc2cn(C)nc2c1 N1(C(COC(C)(C)C(F)(F)F)=O)CCN(C(C2CCCC(F)C2)=O)CC1CCO Cc1nc(NCc2ccnc(OC(C)C)c2)cc(=NCc2ccc3occc3c2)[nH]1 c1(C2N(C(c3ccc(C)nc3)C(=O)NCCOC)CC(O)C2)ccc(C)c(C)c1 CC1CC(C(C(=O)NCC2CCOC2)N(C)Cc2cocn2)CC(C)C1 CC1=C(C)CC(C)(CN2CCCCCC(C(=O)N=c3ccn(CCF)[nH]3)C2)CC1 N1(C(c2ccc(C(C)O)cc2)=O)CCC2CN(C(=O)CC3CC3CO)CC2C1 N1(CC)CCOCC1C(=O)NC(c1cn(C2(C(N)=O)CC2)nn1)C c1(CN2CC(NC(=O)CCc3ccsc3)C(F)C2)cc(Cl)c(F)c(Cl)c1 C12(NC(c3nc(OCC)sn3)=O)CCCC1CN(C(=O)C=Cc1cccs1)C2 C1(NC(CC=CC=C)=O)CCOC(C2CCN(C(=O)CCN(C)CCC)CC2)C1 C1(C)(CNC(CC2C3CN(C(c4nc(COC)oc4)=O)CC32)=O)CCC(O)CC1 CC1CN(C)C(C)CC1NC(C1(C)C=CCN1C(C1CN(C2CCC2)C1)=O)=O c1(C(N2CCCC(C(C)(C)C)C2)C(=O)NCC)cnc(OC)c(F)c1 N1(C(c2ccc(CC)o2)=O)CCCC(C(C)C)(CNC(=O)COc2ccsc2)C1 c1(C(N2CC(CNC(C3CC(OC)C(OC)C3)=O)OCC2)=O)cnc(Cl)c(N)c1 N1(C(CCc2cc(C)nn2C)=O)CC(NC(=O)C2=CCCSC2)C2(CC2)C1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2CCC1C(NC(=O)C=C1CCC(C)CC1)C2 N1(C(C2C(OC)C2)=O)Cc2[nH]nc(C(=O)NCc3ccn(C(C)C)n3)c2C1 C1(C(N(C)Cc2c(C)occ2)=O)CC2(CC(NC(=O)Cc3ccon3)C2)C1 C1(CC(=O)NCC(C)CNC(=O)CCCN2CCCCC2)OCCCO1 c1(C(=O)NC(C(C)NC(=O)CC23COC(C)(C2)C3)C)ccc2ccn(C)c2c1 C1(C#CC(=O)NCCC(C)NC(=O)CC(C)(C)C)(CC)CC1 c1(C(N2CC(NC(CCn3c(C(C)C)ncc3)=O)C2)=O)cn2c(Br)cccc2n1 CCC(CNC(=O)CN(C1CC1)CC)(CC)C(=O)N1CCN(C2CC2)CC1 C1(NC(CCCOC(C)C)=O)CN(C(c2cnn(CCO)c2)=O)CC2(CCC2)C1 C(C(C(=O)NCC(O)CCC1CC1)NC(c1cc(CC)[nH]n1)=O)OCC CC1(C)CCC2(CC1)CC2C(N1CC(Cn2cc(CO)nn2)C1)=O CC1CN(C(=O)C(C2CCCCC2)O)CC(C(=O)N(CCCCCO)C)O1 CCCCC(C)CCC(=O)N1CCCC1C(C)(C)NC(=O)C(c1ccc(C)o1)C c1(C(Cn2cc(-c3ccnc(C(=O)O)c3)nn2)=O)cc(COC)c2c(c1)CCC2 c1(CCC)ccccc1C(=O)NC1CC(C)N(C(c2cc(OC)no2)=O)C1 c1(N2C(C(=O)NCc3nc(C)sc3)CC2)ncnc2cc(F)ccc12 C1(C(N2C3CN(C(c4cnc(C)[nH]4)=O)C(C3)C2)=O)CC12CCOc1ccccc12 C(=O)(CC(C)CNC(=O)C(C1CCCO1)NC(c1cnc(C(C)C)o1)=O)OC C(C(F)(C(=O)N1CC(C)(C(F)(F)F)C1)C(C)C)NC(COCC#C)=O N1(C(C(C)OCCC=C)=O)CC(C)C1C(=O)NCCc1cncn1C C(N=c1ccnc[nH]1)C1CCN(C(c2cncnc2C2CC2)=O)CC1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(NC(=O)C(c2cccnc2)C)CC1 CC1(C)CCCCC1C(=O)NCC1(F)CCC(CNC(c2ncccc2Cl)=O)C1 C1(CC(=O)N(CC(C)CNC(c2ccncn2)=O)C)CCCCCCC1 c1(C(C)CNC(=O)NC(c2noc(CN(C)C)n2)C)cccc(F)c1 C(C)(CC(=O)NCCCn1cc(CC(C2CCOC2)C2CC2)nn1)OC C1(C(=O)NCC(CC#C)(C)C)CCN(C(c2cnnn2CC)=O)CC1O c1(C(=O)NCC2(F)CC(NC(c3cnc(N(C)C)s3)=O)C2)ncc(Cl)cc1Cl C=CCCCC(=O)OC(c1ccc(C(F)(F)F)cc1)C(=O)OC(C)(C)C CC1c2cc(F)ccc2CCN1C(=O)CC(N)C(=O)O C1(C(N(C)Cc2nc[nH]n2)=O)CCCN(C(=O)Cn2cc(C3(C)CC3)nn2)C1 C1(CC=C)(C(=O)NCCCOCC)CCN(C(=O)C=CCCC(C)C)C1 C1(C(=O)NC(C2(O)CN(C(CC3ON=C(CC)C3)=O)C2)C)CCC2CC1C2(C)C C1(CC)CCCCC1C.c12cc(c(C)o1)C(=O)NCC13CC(C1)(C3)NC(=O)CC2 C1(C(=O)NCCCN(CCC)C(c2ccnc(CC)c2)=O)CC1C1CCCC1 C1(NC(C=CC(C)(C)SC)=O)COCCC1SC1CC1 C1(NC(Cc2ccc(C)cc2C)=O)CCCCCN(C(c2cn(C)c(O)n2)=O)C1 C1(C)(NC(c2cnc(C)[nH]2)=O)CCC(NC(=O)C(N2CCCCC2)C)CC1 C(=O)(CC(C)C(F)(F)F)NC(=O)C(N)=O.c1(C2CCC2C)cnccc1C(F)(F)F CC(Cn1cnnc1)N=c1[nH]c(=NCC(C)c2cnc[nH]2)[nH]c2cc[nH]c12 O=C1CSc2ccc(C(=O)NC3CN(C(c4cnsc4)=O)C4CC34)cc2N1 C12(CF)COC(C(N3CC(OC)C(CNC(=O)CC4COC(=O)C4)C3)=O)(C1)C2 C=C1CC(C)(C(=O)NC2CCC2CNC(=O)Cc2cnc(C)s2)C1 C1(CNC(c2c(CC)cco2)=O)CC(C)N(C(=O)COC(C)CC)C1 c1(C(=O)NCCNC(c2cc(C(N)=O)[nH]c2)=O)ccc(S(=O)(=O)C2CC2)cc1 CC1CCC(C(=O)Nc2cccc(CCO)c2)N1C(c1cccc(CCF)c1)=O CC1CC(NC(=O)CCN2CCCCC2CO)CN(C(=O)CN2CCCC2)C1 C(C)(C)(CN=c1[nH]c(N2CCC(CO)C(C)C2)nc2c1CSC2)OC(C)C c1(C(=O)NC2CCN(C(c3c(C)n(C)nc3)=O)CC2O)ccc2ncccc2n1 c1(C(=O)NC(C(C(C)C)Nc2c(C)cnc(C)n2)C)cnc2ccnn2c1 C(=O)(CC(C)(O)C(F)(F)F)N(CCCCN(C)C(c1ccc(O)nc1)=O)C C1(C(=O)NCC(C)NC(c2csnc2C)=O)CCN(C2CCSC2)CC1 CC1CC(CNC(C2CC(O)(C(F)(F)F)C2)=O)CN1C(C1CC(F)(F)C1)=O c1(C(=O)NCC(C)NC(=O)CCn2cncn2)csc(C2CCCO2)n1 N(S(=O)(=O)N1CCC(C(=O)NNc2ccc(C(N)=O)nn2)C1)C(C)C1CC1 C1(SCC)CCC(C(=O)NC2CCN(C(c3ccc(C(F)(F)F)[nH]3)=O)C2C)CC1 c1(C(=O)NC2CCN(C(c3cncc(OC)c3)=O)CC2F)ccc2sccc2c1 N1(C(C(C(=C)C)(C)C)=O)CC2CC(C1)CN(C(=O)CSCCN(CC)CC)C2 C1(CC(=O)NCc2cn(Cc3cccc(C(F)(F)F)c3)nn2)CCCC1(F)F N1(C(c2nnn(C(C)(C)C)n2)=O)CC2CC2(NC(=O)Cc2cnccn2)C1 N#Cc1ccc(C=CC(=O)NCC2(CNC(c3ccc(F)o3)=O)CC2)cc1 Cn1cc([N+](=O)[O-])cc1C(N1CCC(NC(=O)CC2CCCCC2O)C(F)C1)=O C1(CCOC)CN(C(c2ccc(C(N)=O)o2)=O)CCN1C(c1ncoc1C)=O C(C)(C(C(=O)NCc1c(CO)noc1C)C(C)C)NC(c1c(C)cccn1)=O c1(C(=O)NC(C2CCCC2)CNC(Cc2ncc(C)[nH]2)=O)cc2sccc2s1 c1(NC(C2(CC=C)CCCN2C(c2csc(F)c2)=O)=O)cc(C)ccc1C Cc1cc(C(N2CC=CC2CNC(=O)C(F)(F)CC2CC2)=O)cc2ccsc12 C(=O)(CCC(C)(C)F)NCCC1(C(=O)NC(c2ccc(F)nc2)C)CCCC1 CCC(O)C(C)C(=O)N1CCC(C)C1CNC(=O)C(C(C)C)OCC(C)C N1(C(CC(C)N(C(C2CN(C)C2)=O)CC)=O)CCN(C(=O)CO)CC1 c1(CCC(=O)N(C2CN(C(=O)Cc3cc(C(F)F)nn3C)C2)C)ccc(O)nc1 CC1(CNC(c2cc(=O)cc(Cl)[nH]2)=O)CCCN(C(c2cc3sccc3s2)=O)C1 N1(C(C)=O)CCOC(C(=O)N(CC(C)CN(C(=O)C=CC2CCCCC2)C)CC)C1 N(C(=NCCS(=O)(=O)N1CCCC1)NC(C)C)C(C)C.c1(CCC)cccnc1 C(=O)(C(F)C(C)(C)O)N1CC(CC=C)(C(=O)NCCSCCC(F)(F)F)C1 c1(C(=O)NC2C(NC(C(C)NC(c3ccco3)=O)=O)C2)c(Cl)ccc2c[nH]nc12 C1(OCC)CCC(NC(=O)C(C)(C)C2CCCN2C(C2CCC2C(C)C)=O)CC1 c1(CC)ccccc1CNC(=O)C(N1CCC(OC2CC2)C1)=O Cc1cc(-c2nc(C3CCOCC3)nn2C2CCSC2)cc(C)c1F N12CC3C(C3C1)CC(=O)NCC1(C)CCCN21.c1(C(CC)OC)ccccc1 C1(C(N2C(CN(C(Cc3c(C)cnn3C)=O)C)CCC2)=O)CC2(CCC2=O)C1 C(CC(=O)NCC(C)(CO)NC(=O)CCc1ncc(C)[nH]1)(C1=CCCC1)OCC C1(OC)CC2CC(C(=O)NC(C3CCN(C(=O)CN4CC5CC5C4)CC3)CC)CC12 C(=O)(C(CC(N)=O)NC(=O)C(O)C(F)(F)F)N(CC(C)N(C)Cc1ccsc1)C C1(C(=O)NCC(C)(C)NC(C2C(CC)C2)=O)(CF)CC(F)(F)C1 C1(CNC(c2cn(CCC)nn2)=O)CN(C(c2cnc(SC)s2)=O)CCO1 Cc1[nH]c(C)c(C(=O)NC2CCC(NC(C3CCCCC34CC4)=O)CC2)c1C C1(O)(CCNC(C2(CC)CCC2)=O)CCCN(C(C2COC3(CCC3)C2)=O)C1 c1(C(=O)NC2CCC(CNC(CC(C)O)=O)CC2)ccc2nn[nH]c2n1 N1(C(c2c(C)cc[nH]2)=O)CCN(C(=O)CNc2ccccc2[N+](=O)[O-])C(C)CC1C C1(NC(C(CC)(F)F)=O)CC2CCC(C1)N2C(c1ccccc1OC(F)F)=O C(=O)(C(C)CC(C)(C)C)N1CCN(C(C2CC=C(C)CC2)=O)C(CO)C1 CC1CC(C(N2CCC(O)(C(N)=O)C2)=O)CN(C(c2cncn2C2CC2)=O)C1 N1(C(C2(NC(c3ncccc3F)=O)CCCC2)=O)CCCC(C2CCC2)C1 N1(C(C(c2cccc(O)c2)C)=O)CCCCC1CCNC(=O)CCF Cc1c(Br)csc1C(N1CCCCC1Cn1cc(-c2cccc(F)n2)nn1)=O c1(C(=O)NC2C(C)CN(C(C3CCS(=O)(=O)CC3)=O)C2)noc2ncccc12 N1(C(CC(c2c(C)noc2C)C)=O)C2CCC1CN(C(=O)C(C)NC(N)=O)CC2 C1(CC(=O)NCC2C(CC)C2)CN(C(C2CNC(=O)O2)=O)CCO1 N1(C(C(CC=C)CC)=O)CC(NC(=O)Cc2cccnc2)CC(C)(C)C1 C1(C(c2cccc(Br)c2)O)CCCN1N1CCc2cc(Br)cnc21 c1(C(=O)NCC(C(C)C)NC(C(CC)NC(C)=O)=O)cc2scnc2[nH]1 CC(C)(CCC(=O)N1CCNC(=O)C1)NC(=O)Cc1ccoc1 c1(SCC2N(CCCCC)CC2)ccc(NC(=O)CCc2ccccn2)o1 C1(C(=O)NC(CCN(C)C(c2ccnn2C2CCCC2)=O)(C)C)CCCOCC1 c1(CCC(=O)NC2(C)CC(NC(C3(F)C(C)C3)=O)C2)cnc2n1CCCCC2 C12(C(=O)NCC3(NC(C4(c5cccc(C)c5)CC4)=O)CC3)CCCC1C2(F)F C#Cc1ccccc1C(=O)NC1CC(C)C1.c1(C(C)C2CC2)ncccc1COC C1(CNC(C2(C(=O)NC)CCC2)=O)CC(O)CN1C(=O)C=C(C)C(C)C C(=O)(C1=NOC(C)(C)C1)NCCCC1N(C(CCCC=C)=O)CCCC1 C1(CNC(=O)COCC(F)F)CCCN(C(=O)CC2(CNC)CCCC2)C1 C=C(C(=O)N1CCOC(CC(=O)Nc2cnc(Br)cc2N(C)C)C1)C(F)(F)F N1(C(COC)=O)CCCCC1CN(C(=O)CCNC(c1cccc(Cl)c1)=O)C C(=O)(CCC(C(=O)NCCC(C)NC(c1cccc2c1OCC2)=O)N(C)C)OC Cc1cc(C)n(CCCNC(=O)C(=O)NCCC2CCCCO2)n1 CC(C)CC(CNC(=O)C#CC1CC1)C(=O)NOCCCF CC1CN(C(C2(P(C)(C)=O)CC2)=O)CC1CNC(c1ccc(CO)cn1)=O C1(NC(c2c(CC)cno2)=O)CS(=O)(=O)CC1NC(=O)CN1CCCOC1=O c1(OC(C(=O)NC(CN(C(C(CC)OC)=O)C)(C)C)C)ccc(Cl)cc1C C(C(C)C(=O)N(C)CC1CN(C(=O)CC2(n3ccnc3)CC2)C1)OC c1(C(N2CC3CC2CN3C(c2cc(Cl)cc(Cl)c2)=O)=O)cn2c(F)cccc2n1 C(C(=O)N1CCCC(N2CCN(C(C3CN(C)C(=O)N3)=O)CC2)C1)(C(C)C)SC c1(OCC(=O)NC(C2N(C(C(F)OC)=O)CCC2)C)ccc(C(C)C)cc1 N(C(=NCC(O)c1cccc(Cl)c1)NC1CC1)C1CC(OC(C)(C)C)C1 CSC1=C(C(=O)N2CC(O)CC2CNC(C2CC2(C)C)=O)CCCC1 C(=O)(C1=C(Cl)CCC(C)C1)N1C2(CNC(C3(COC)CC3)=O)CCCC(C1)C2 C#Cc1c[nH]nc1C(=O)NCC(CC1CCCC1)C(=O)NCC(C)CCO c1(C(N2C(C)CC(CNC(C(C)=C(C)C)=O)C2)=O)ccc(CO)cc1F C(CC(F)F)(C(=O)NCC1CCCC1(C)C)NC(C(C)n1cccn1)=O CC1(C)CCC(CNC(C2(NC(C3CN4CCC3C4)=O)CC2(C)C)=O)C1 C1(CNC(C(N2C3C(NC(N)=O)C(C3)C2)=O)=O)C2CCCCCC12 N1(C(c2cc(CC(C)C)on2)=O)CCCN(C(=O)C2=CCC(C)CC2)CC1CO S(=O)(=O)(c1c[nH]c2cc(Br)cnc12)N1CC2C(N(c3ccccc3)C)C2C1 c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(CC)o2)=O)ccc2c(c1)CCCC2 CCC(C(=O)NCCC(O)CNC(=O)CCn1cccn1)C(C)C C1(CCC=C)CCCCN1C(c1csc(C(C)(F)F)n1)C(=O)NCCCF c1(C(=O)NCCO)cnncc1C(F)(F)F.C=CCC(=O)NCCCCC=C(C)C C1(NC(=O)C(F)=CC2CC2)CCN(C(c2cnc(C3CC3)s2)=O)CC1F C1(C(=O)NCc2ccc(O)cc2F)CCC2CCC1N2C(=O)C(O)C(F)(F)F c1(CNC(C2C3CCCCC23)=O)cccc2c1CN(C(=O)C=Cc1nccs1)C2 C(=O)(N=c1cc(Br)[nH][nH]1)c1cccc(Nc2nccc(C)n2)n1 C1(C(=O)OC(C(=O)NC(C2(CO)CC2)C)C)CC1[N+](=O)[O-] c1(CC)nc[nH]c1C(=O)NC1CCC1NC(=O)CCSc1nccn1C C1(C(N2CCC(CN(C(C3CN(CC)C(=O)N3)=O)C)C2)=O)CC12CCOC(C)C2 N1(C(c2nccc(C(N)=O)c2)=O)CC(NC(=O)CCCC2CCC2)CC12CCC2 c1(CC(=O)N(CCCNC(c2c(CC)cno2)=O)CC)c(Cl)cccc1Cl N1(C(CCCC(=O)NCCC)=O)CCC2C1CCCN2C(=O)C(C)OCC(F)(F)F c1(C(N2CC(C(=O)NC3=CN=C3NC(C(C)(C)OC)=O)C2)=O)ccc(Cl)c2occc12 C(=O)(NN1C(=O)CCC1C)c1cnn(C(CC)C)c1C c1(C(N2CC3(C(NC(C(C)OC)=O)CCC3)C2)=O)cccc([N+](=O)[O-])c1O c1(C(N(CCCN(C)C)CCNC(C(CC=C)C)=O)=O)cnc2c(c1)COC2 c1(C(N(CCC(C(C)C)NC(C2(CO)CC2)=O)C)=O)cc(F)c(F)cc1F C(C1CCOCC1)=CC(N1CC(NC(CN(C)CCNCc2ccoc2)=O)C1)=O CCCC(C#N)C(=O)N1CCC(Cn2cc(-c3cnn(C)c3C(C)C)nn2)C1 C1(C(C)=O)CCC(C(=O)NCC2CCN2C(=O)CC(=O)OCCC(C)C)CC1 N1(C(C(CC#C)C)=O)CCC(F)(F)C(CNC(=O)CC(=O)NCC(F)(F)F)C1 c1(C(N2CCC(CC)C2CNC(=O)CCCNC(N)=O)=O)[nH]ccc(=O)c1C C1(CC)(CC)CC(NC(=O)CC2C=NN(C)C2=O)CN1C(c1cc[nH]n1)=O CC1COc2ccccc2C1C(=O)NCC1CCN1C(C12CCC(CC1)OC2)=O N1(C(C=C(CC)C)=O)CCN(C(C23CCCC(C2)OC3)=O)CC1c1ccccn1 c1(N(C)CC2(CC(C)C)CC2)nc(=NC2CSC(C)C2)[nH]c2ncn(C)c12 c1(OC)cc(OC)cc(C(=O)NC2CN(C(c3ccn(C)n3)=O)CC2F)c1 CC1=C(C(=O)NCC2CC(NC(=O)CCC3CCCC(=O)N3)C2)CCCC1 c1(NC(C2N(C(C#CC)=O)C3C(C2)C3)=O)cc(Br)c(C)c(Br)c1 N1(C(CC=CCNC(C2(C)CCC2)=O)=O)CC2(CCC(CO)O2)C1 N(C1CCCn2nccc21)C(C(C)NC(=O)COc1ccc(Cl)c(F)c1)=O c1(CC)cccc(NC(C2(N(C(=O)C=CCC3CCC3)C)CC2)=O)c1O C(CC(=O)NC(Cn1cncn1)CC)(C(F)F)NC(CCCOC(C)=O)=O C(C(C)(O)C(=O)OC)NC(CN(C(=O)CCc1ccn(C)c1)CC#C)=O CC(C)C(CNC(=O)COC1CCCCC1)NC(c1ccsc1C(F)(F)F)=O N(C)S(=O)(=O)N(C)C.Cc1cc(OCC(=O)NC(C)CN(C(=O)C(C)(F)F)C)no1 N1(C(c2c(O)ncc(N(C)C)c2)=O)CCC2CN(C(=O)C(C)(C)CF)CC12 Cc1nnc(C(=O)NCC(F)CNC(=O)C(C)OC(C)(C)C)s1 N1(C(C(C=C)(C)O)=O)CCN(C(c2ccc[nH]2)=O)C(c2cc(F)ccc2F)C1 C1(C2CN(C(c3nc(CC)sc3)=O)C2)CCCCN1C(C1OCCC1C(C)C)=O C1(NC(C2CC(CCO)C2)=O)CC12CCN(C(=O)CN1CC3CC3C1)CC2 CCC(C)CCC(O)CC(=O)N(C)CCN(C(=O)CC1CC1)C(C)C c1(OC(C)=O)ccc(NC(C)CCN(C(=O)C(=O)N(C)C)C)cn1 C1(CNC(C2CC(C)(F)C2)=O)(CNC(c2ccc(C3CC3)cn2)=O)CC12CCC2 N1(C(C23CCC(OC)C2C3)=O)CCC=C(CNC(c2cc[nH]n2)=O)C1 CN1CC(C(=O)N(CCCNC(c2ccc(C(C)(C)C)o2)=O)C)C(C(F)(F)F)C1 C1(CC=C)(NC(=O)CC(=O)NC)CCCN(C(C2OCCN(C)C2=O)=O)C1 c1(C(N2CC(CNC(C3CC=CCC3)=O)C2)=O)cc2nccc(C(F)(F)F)n2n1 Cc1cc(NC(C2C3COCC23)=O)c(C)cc1F c1(CC(=O)NC(CCNC(c2c(C(=O)OC)cn(C)n2)=O)C)cc(C)nc(O)c1 N1(C(C2=CCN=N2)=O)CCC2(CCN(C(C3CCC(C)(C)O3)=O)CC2)C(C)C1.CO C1(NC(C2CC(C)N(C(=O)CC(=O)OC(C)(C)C)C2)=O)CC2CCC(C1)S2 CCC1=NOC(C(N2CCCC2C2CCN(C(=O)Cc3cc(C)sc3C)C2)=O)C1 C1(NC(CC2CC(=C)C2)=O)CC(C(=O)NCCC(O)CC)C12CCC2 N1(CCSc2n(C(C)C(=O)O)ncn2)CCC(NC(=O)OC(C)(C)C)C(C)(C)C1 c1(C(N2C(CN(C)C(C3C(F)(F)C34CCC4)=O)CCCC2)=O)ncc(Cl)nc1Cl c1(CC=C)cnc(C)c(OS(=O)(=O)Cc2ccccc2OC)c1.C1(=O)C(C)O1 N1(C(C(=O)OCC)=O)CCCN(C(c2ccc(OC)c(C(F)(F)F)c2)=O)CC1 c1(OC)cncc(C(=O)NCCC2(NC(c3cnc(C(C)C)s3)=O)CCC2)c1C Cc1ncc2n1CC(C(=O)NCC1COCCN(C(=O)Cc3n[nH]c(=N)s3)C1)CC2 C1(CNC(COCCCOC)=O)CN(C(=O)C=CC=C(Cl)Cl)CC1C CN1CCCC(O)(CC(=O)NCC2CN(C(c3cn(C(F)F)cn3)=O)CCO2)C1 C(N=c1[nH]cnc2c1CCC2)C1(CNC(C(CC)OCC)=O)CCC1 C1(NC(CC(=C)I)=O)CCSC12CN(C(c1ccon1)=O)C2 Cn1c(C(=O)NCCNC(=O)C(F)=CCCF)cc2cc(Cl)ccc12 C(=O)(C(O)C(C)(C)C)OC.C12(CNC(=O)C1)c1cn(nn1)C1C(CCCC1)CN2 C(=O)(C(=O)C(F)(F)F)NC1CN(C(C=Cc2ncn(C)c2)=O)C1 C1(C(N2CCC(CCNC(=O)CSC(F)(F)F)C2)=O)CC2CCC(C1)O2 C1(NC(c2cc(CO)on2)=O)CCC2(CCN(C(c3cnn(CCF)c3)=O)C2)C1 C1(C(=O)NC(CC(C)NC(c2cncc(F)n2)=O)C)CCCC(F)(F)C1 CC1CN(C(c2coc(Br)c2)=O)CCN1C(c1coc(CC2CC2)n1)=O C1(C(N(C2CCCN(C(=O)C(C)(C)C3CC3)C2)CC)=O)CCc2ncccc2C1 c1(OC)ccc(S(=O)(=O)NCCCc2nc(C(C)(C)C)no2)c(F)c1F N1(C(C(=O)OCC)=O)CCC2(CC1)CN(C(=O)C(C)CS(C)(=O)=O)CCC2O Cc1ccnc(CNC(=O)C=CCN(C)C(c2cnsc2)=O)c1 CC1=NS(=O)(=O)NC=C1C(=O)N1CCC(NC(c2cc(Cl)ccn2)=O)C1 CCCC(C(=O)NCC=C1CCN(C(c2ncc(Br)cn2)=O)CC1)OCC C(CCC(C)CO)NC(COCCNC(c1ccc(C(=O)OC)[nH]1)=O)=O N1(C(CC=CC)=O)CCC2CC1CN(C(=O)Cc1ccc(OC(F)(F)F)cc1)C2 C1(NC(C2CCCN(C)C2)=O)CCN(C(c2cccc(C3CC3)c2)=O)C12CC2 C1(C(N2CC(CN(C)C)C2)=O)(NC(=O)Cc2nccn2C)CC(F)C1 C(CCCCC(=O)NCCCN(C)C(C)=O)N(C(C(C)OCC=C)=O)C C(CNC(c1ccnn1CCF)=O)(C(=O)NC1(C2CCCO2)CC1)SC CC1CN(C(c2cccs2)=O)CCC1CNC(=O)COc1cccc(Cl)c1Cl c1(C(N2CCC(C(=O)NC(CC)CC)C(O)C2)=O)cc(Cl)cc([N+](=O)[O-])c1C C(=O)(CCCCC(F)F)NC(C(C)C)CCNC(=O)C(C)(C)C(F)F C(=O)(CCC(C)(C)C(=O)NCCC(C)CCNC(c1csc(COC)c1)=O)OC c1(C(=O)NCC2(NC(C3C(C=C(C)C)C3(C)C)=O)CCC2)nnn2c1CSCC2 N1(C(C(C)(C)c2ccccc2)=O)CC2(CCCC2)C1C(N1CCOC(=O)C1)=O n1(C(C)OCC)nc(Br)c(CNC2(O)CCN(c3ccccc3)C2)c1Br C1(C(=O)NCCN(c2ncnc(Cl)c2F)CC)CN2CCC1(C)CC2 N1(C(c2cc(C)on2)=O)CCCC2CCN(C(c3cn(C(C)C)cc3C)=O)CC12 N1(C(C2N(C(C)C)CCC2)=O)CC2CN(Cc3c(F)cccc3C#N)CC2C1 N1(C(c2ccc(CC)cn2)=O)CCC(NC(c2ccccc2C)=O)C(F)C1 C1(NC(C(C)C2CCCC2)=O)CCC(C)N(C(c2cnn(C)c2Br)=O)C1 N1(CC)CCCC(C(N2CC(CNC(=O)C(CCOC)N(C)C)C2)=O)C1 C12(C(=O)NCC(CNC(C3=NOC(C(C)(C)C)C3)=O)CO)CC=CCN1CCC2 O=C(C#Cc1ccccc1)NC1CCCN(Cc2nccc3ccccc23)CC1 CCCCC(O)C(=O)NCCCCNC(C1(C(C)(F)F)CCC1)=O N1(C(c2c(OC)cnnc2OC)=O)CCC2(CCN(C(C3CC=CCC3)=O)C2)C1 C12(CNC(C=CC(CC)C)=O)CCCC1N(C(=O)COC1CCCC1)CC2 Cc1cc(CCC(=O)NCC2C=CCN2C(=O)CC2CCCC2)nn1C n1(CC(N2C(CNC(=O)CC3CCCCC3O)CC2)=O)c(O)nc2ccccc12 C1(NC(C2(COC)CCCCO2)=O)CC(C)CN(C(=O)C(N)=O)C1 C1(C2CCCC2)(NC(CCC2CCC(C)O2)=O)CC1.C12CCN(C1)C2=O N1(C(C2(C=C)CC2)=O)CC2=C(C1)CN(C(c1cc(C)c(C)o1)=O)C2 C(=O)(C(CC)C(=O)OC)N1C(NC(c2nc(OCC)oc2)=O)CC(OC)C1 C(=O)(C1=CCCOCC1)NCCC1CCN(C(=O)CSc2ccc(F)cc2F)C1 O=S(=O)(c1nc2c(s1)CCCC2)NCc1ccc(OC(F)(F)F)cc1F Cc1c(C(N2CC3CCC2CN3C(C2CCO2)=O)=O)[nH]c2ccccc12 CC(C)CCCOCC(N1CCCC1CC(=O)NCC(O)(CO)C1CC1)=O Cc1cc(C(=O)NC2CCCC2NC(C2CC2C(N)=O)=O)c(C)[nH]1 Cc1nc(Nc2cnn(C3CCCCO3)c2)ncc1Br C1(NC(c2n(C)nc(Br)c2)=O)CN(C(=O)CCCC(=O)C2CC2)CCC1CO c1(CC)c(C(=O)NCC2CC(C)N(C(=O)C=NOC)C2)cnn1CC c1(C(N2CCCC(CCNC(C3=CC(C)CC3)=O)C2)=O)onc2c1CCCC2 N1(C(c2c(N)non2)=O)CC(NC(=O)CNC(c2ccco2)=O)C2CCCCC12 c1(C(N2CC(O)(CN(C(C(C)C#N)=O)C)C2)=O)nccc(Cl)c1F C12(C(=O)NC3C(NC(C(CC)C)=O)CCCC3)CC3CC1C2C3O C1(CNC(C(=O)NCCOC)=O)C(C)CCCN1C(=O)CCC(F)F C1(C(=O)NCC(CC)(C)NC(=O)Cc2c(C)n[nH]c2C)CC(N=[N+]=[N-])C1 C1(CNC(CC(C)c2ccncc2)=O)CCCCN(C(c2cn3ccnc3s2)=O)C1 n1(CC)nnc(C)c1C(=O)NCCCC1CN(C(=O)Cc2n[nH]c(=N)s2)CCO1 C1(Cn2cc(CC(C)(C)OC)nn2)CCCN(C(=O)CC(O)c2ccccc2)C1 C1(NC(CC=C(C)C)=O)CCN(C(C2C=CC=CC=C2)=O)CC1CO C12(NC(=O)Cc3cscn3)CCCC1(F)CN(C(C1(C(N)=O)CC1)=O)C2 C(=O)(C(CNC(=O)CCCC)CC(C)C)NC(C#C)(CO)CO CCS(=O)(=O)C=CC(=O)NC1COCCN(C(C2SC3C=CC2CC3)=O)C1 c1(NC(CCC(N2CCC(O)(N(C(C)=O)CCF)C2)=O)=O)ccncc1F c1(C(=O)NC2C3CN(C(c4cncn(C)c4=O)=O)CC32)c[nH]c2cccc(Cl)c12 S(=O)(=O)(c1ccccc1C(N)=O)N1CC(C)(C(=O)Nc2cccc(CC)c2O)C1 c1(-c2c(C(=O)OC)cncn2)cnn2ccc(C)cc12 C1(CNC(C(C)=C2CCC2)=O)N(C(=O)CC2CC(C)(C)CO2)CCCC1(C)C c1(C(N(CCCNC(=O)C(c2ccccc2F)C)C(C)C)=O)ncc(F)cc1N c1(C(=O)NC2C(NC(C(CCC)N(C)C)=O)C2)c(C(C)C)cccc1F C1(C(=O)NCCCOC)CC2(C1)CN(Cc1ccc(C)cc1)C2 N1(C(c2cc(OCC)no2)=O)CC2CCOCC2(NC(=O)C2=CCOC2)C1 CC(CC(=O)NCC(C)(F)CNC(c1ccc(=N)[nH]n1)=O)C(F)(F)F N1(C(c2c(OC)ccc(Cl)c2)C(=O)NC(C)C)CCc2ncn(C)c2C1 c1(C(=O)NC2C=CCN(C(C=C(CCC)CCC)=O)C2)cnc2ncccc2c1 CC1CN(C(c2cn[nH]c2)=O)CCN1C(c1csc(-c2ccccc2)n1)=O c1(C(N2C(CC)C(NC(C3CCC4CCC34)=O)CCC2)=O)ccn2ccnc2c1 C1(NC(=O)Cn2cnc(C(F)(F)F)n2)CCN(C(C2CCCCC2O)=O)C12CC2 N1(C(CSCC(=O)OC)=O)CCC(C)(C)C(NC(=O)CC(=C)C)C1 C(=O)(CCC(F)(F)C(F)F)NC(COC)CNC(=O)C1=CC(C)(C)C1 C1(C(C)NC(c2ccsc2)=O)CCCN(C(=O)COCCCF)C1 C1(C(=O)NCC2CCCCO2)CCC2(CC2)N1C(c1cc(F)c[nH]1)=O C1(C(N2CC(CNC(C3CC4CCC3CC4)=O)C(O)C2)=O)CC12CCOCC2 c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)Cn3cncn3)C2)c1 S1(=O)(=O)c2ccc(c(Br)c2)CN1.CCCC(CCC)C1C(SCC)CCCC1 C(CC(C)(C)C(=O)N(CCC(=O)N(C)C(c1ccccc1)C)C)OC C(CNC(=O)CCn1cc(CCCOC(=N)O)nn1)(C(C)C)OCC C1(CC(=O)NCC2(O)CC(CO)C2)COCCN1C(C1COCOC1)=O C1(NC(c2cccc(C)c2F)=O)CN(C(=O)CCN2CCC2)CC1N=[N+]=[N-] c1(OC)cc(Br)cnc1C(N1CC(NC(C2(CC3CC3)CCC2)=O)C1)=O C#CC1CN(c2cc(C(=O)O)cn(C)c2=O)CCN1C c1(C(=O)NC23CC(NC(c4ncn(C)n4)=O)(C2)C3)sc2sccc2c1Cl N1(C(CC(COC)C)=O)CCCC(F)(C(=O)NC2CCCCCC2OC)C1 Cc1cccc(CC(N2CCOC(CNC(=O)COC3CCCCCC3)C2)=O)c1 c1(NC(CNC(C(=O)OC)C2(C)CC2)=O)nc2ccc(C)cc2[nH]1 C(=O)(CCCC(C)(C)NC(C1CC1F)=O)NCc1ccc(OC)cn1 C#Cc1ccc(Cl)c(C(=O)NCC2CN(C(=O)C(C)SC)CC(C)(C)O2)c1 CC(F)(F)CCCCN=C(NCC1(S(C)(=O)=O)CC1)NCC(F)F Cc1cc(C(=O)NC(C(=O)NCC(C2CCCCO2)O)C2CC2)sn1 N1(C(=O)CCSc2ccc(Br)cn2)CCN(Cc2cccnc2)CC1 N1(C(C(C2CCOC2)OCC)=O)CC2(C1)CN(C(=O)C(C)(COC)COC)C2 c1(SC)ccnc(N2CC3C(CNC(c4ccnc(CO)c4)=O)C3C2)n1 c1(C(=O)NCC(CCNC(c2nc(CC)oc2)=O)O)oc2ccccc2c1Cl CC1CCNC1C(=O)NCCCCn1ccnc1 c1(NC(C(=O)Nc2c(C)nn(C)c2)=O)ccc(SC2CCCCC2)c(F)c1 C[S+](C)CCC(O)C(=O)NCCCNC(c1c(F)ccc(F)c1N)=O C1(C(=O)NCCC(C)(C)NC(CCC2CC(OC)C2)=O)CCc2nnnn2C1 N1(C(c2n(CCC)ccc2)=O)CCC(CO)(CNC(C2(C)CCOC2)=O)CC1 C1(O)(CN(CC(C(=O)NCCC)F)CC)CCN(C(C2CC=CCC2)=O)CC1 C(CCCC(=O)OC)(c1n(CCCNCc2ccc(Cl)c(C)c2)nnn1)OC C(=O)(CCC(=O)N(CC(C)NC(C1OCCC1C(F)(F)F)=O)C)OCC c1(CC2(C(=O)NCCCC3CC3)CN(C(CC)=O)C2)ccc(Cl)cc1 N1(C(c2cc(C)nn2C(F)F)=O)CCC(NC(c2scc(C)c2Cl)=O)C(F)C1 C1(C)(C(=O)OC(c2ccc(C)[nH]2)C)CC2CC2C1 O=C(C1=CC2CC(C1)CC2O)NCCC1COC(C(F)(F)F)CN1C(=O)C1CC1 c1(C(N(C(CCNC(C2(OC)CCCOC2)=O)C)C)=O)cnc(N)c(Cl)c1 CC1(C)CC=C(C(=O)N2CC(C(=O)NC3CCC3O)C3(CCC3)C2)CC1 c1(C(C(=O)NC(C2CCN(C(=O)C=C3CCC3)C2)C)C)ccccc1F N1(C(c2c(C)nc(CC(C)C)o2)=O)CC2CCC1CN2C(=O)C(F)CC(C)C C1(NC(C(C)C)=O)CCN(C(C2COCCN2C)=O)CC(O)C1 C1(CC(=O)NCC2=C(C)CCC2)CN(C(=O)C(C2CC2)OC)C(C)(C)C1 C1(CC(N2CCC(F)(CNC(c3cc[nH]n3)=O)C2)=O)COC2(CCC2)CO1 C(C(C)(C)CCCNC(=O)OC(C)(C)C)N(C(C(C)CN1CCOCC1)=O)C C12(NC(c3n(C=C)nnc3)=O)CCC1CN(C(=O)C=C(C)C1CC1)C2 Cc1nn(C)c2c(N3CCC(CC(F)F)C3)nc(N3CCC(=O)N(C)CC3)nc12 C(=O)(CCC(F)(F)CN=[N+]=[N-])N(C1CCN(C(c2cnc(C)o2)=O)C1)C CC1CCC(=CC(=O)NC2CCN(CC(F)(F)F)C2)CC1.c12cn(nn1)CNC2=O C(=O)(CCCCC#N)N(C(C(=O)NCc1nc(C)c(C)o1)C1CC1)C c1(N(CCOCCOCC)C)cccc(NCC2(C(=O)O)CCCOC2)c1 CCS(=O)(=O)NCCNC(=O)C(C)NC(C1CC(OCC)C1)=O CC1=CC(C)C(c2c[nH]nn2)CC1.C(CCC(C)(C)C)C1CCN(C)N1 C(=O)(CC(CC(=O)OCC(C#C)CC)NC(=O)OC(C)(C)C)OC C1(NC(c2c(C(C)C)cc(F)cc2)=O)CCN(Cc2cccnc2)C1(C)C Cc1ccc(C(=O)NC(C)C(CO)NC(=O)C(O)C(F)(F)F)c(C2CC2)c1 c1(C(=O)NCCC)ccccc1OC1(CO)CN(C(c2ccsc2CC)=O)C1 c1(C(C(=O)NCC2N(C(CCC(C)N(C)C)=O)CC2)=O)cc(F)c(F)cc1F C1(C(N(CC(=O)NCC)C)=O)C2CCN(C(=O)C=C(C)COC)CC12 C1(NC(C(C)C2CCCC2)=O)CCC(C)(NC(c2ccncn2)=O)CC1 C1(C(N2CCC(CNC(c3cnco3)=O)C23CCC3)=O)CC2CCCCCCC12 Cc1nccc(C(=O)NCCCN(C(=O)C(C#N)C(C)C)C2CC2)c1C Cc1nc(C(N2CCC(CC3(C(=O)N(C)CC4CCCOC4)CC3)C2)=O)n(C)n1 C1(CNC(c2cccs2)=O)CC2CCC1N(C(=O)C(O)C1CC1)C2 N1(CC(=O)NC(C2CC=CCC2)C(=O)N(CC(C)C)CC)CCCC1CSC c1(C(N2CCN(C(c3cc(Cl)cs3)=O)C(C)C2)C)ccc(Br)cc1F C1(C(=O)O)CC2(CCC2)CN1C(c1csc(Cc2ccc(Cl)cc2)n1)=O N(C(=NCCc1cccnc1)NCC1CCSC1)C(c1ncccc1F)C Cc1c[nH]c(C(N2CC(C(C)(C)O)(CNC(C3CCN3S(C)(=O)=O)=O)C2)=O)c1 C#CC(CNC(c1coc(C(C)NC(C2(C(C)(F)F)CC2)=O)n1)=O)CC1CC1 N1(C(C2CN(C(C(CCCC)F)=O)C(C)CC2)=O)CCC(C2CCOC2)C1 N1(C(c2nnc(C)s2)C(=O)NCCC#N)CCOC(CN(C)C)C1 N1(C(c2c(CC)nccc2)=O)CCC(C(=O)Nc2ncccc2CSC)C(O)C1 N1(C(CCC(CC)C)=O)CC(NC(c2cc(C(C)(F)F)n[nH]2)=O)CC2(CC2)C1 c12ccc(cc1)[nH]2.N1(N(C)C(=O)NCc2c(C)noc2)CCC(C)CC1 c1(C(N(CCOCCN(C(C2(OC)CC2)=O)C)C)=O)ccc(C)c(NC(C)C)c1 N1(C(C=CC=CCC)=O)CCOC(C(N2CCN(CC(C)O)CC2)=O)C1 Cc1cccc(C2C(C)CN2CCCC(=O)NCC(C)C)c1 n1(CC(=O)NCC2CN(C(C3CCCC3)=O)CC2C(F)(F)F)ccc([N+](=O)[O-])n1 Cn1ncc([N+](=O)[O-])c1C(=O)NCc1cccc(CNC(=O)CCCN=[N+]=[N-])c1 C=CCCCCN(C(=O)CN(C(=O)C(CC1CCCC1)OCC)CC)C CCC(CC(=O)N1CCCCC1CC(=O)NOCC(C)(C)O)OC CC1CC(C)(C(N2CCC3(CC2)CC3C(=O)N2CC(O)CCO2)=O)CC(C)O1 N1(C(c2n[nH]c(=N)s2)=O)CC2CCCC(C1)N2C(c1ccncc1)=O C12(NC(C3C(=C)C3)=O)CCCC1N(C(c1cccc(-c3nc(C)cs3)c1)=O)CC2 N1(C(c2cccc(OCC)c2)=O)CCC(NC(c2ccno2)=O)C(C)(C)C1 c1(C(N2CC(NC(c3cncc(-n4cccc4)c3)=O)C2)=O)cc2n(c1)CCCC2 N1(C(C(COC)OC)=O)CCC(C(=O)NCC2(F)CC(CO)C2)C12CCC2 c1(C(=O)NCC2N(C(C3CC(OC)C3)=O)CC(C)CC2)nc(C)c(C)[nH]c1=O c1(C(N(C2CCN(C(C3=C(C)OCC3)=O)C2)C)=O)ccc2scc(C)c2c1 N1(C(C2(CC#C)CCN(C(C3CN(C(N)=O)C3)=O)C2)=O)CCCC(O)CC1 n1(CCOC)ccc(=NC(=O)CCCCCN(C)C(C2C3CCC(C3)C2C)=O)[nH]1 C(=O)(CC(C)(C)CC(F)F)CC1C(NC(c2c(NC(C)=O)nc(Cl)cc2)=O)CC1 c1(SCC)ccc(C(N2CCCC(CCNC(C3(NC(C)C)CC3)=O)C2)=O)cc1 O=C(Cc1ccccc1Br)N=c1cc(CCNc2cnco2)[nH][nH]1 c1(C(=O)NC2C(NC(c3ccc(OCC4CC4)cc3)=O)CC2)ccccc1F C1(F)(CNC(C2C(C)(Br)C2)=O)CC(NC(=O)COCC(c2ccccc2)C)C1 N1(C(CC(CC)(F)F)=O)CCC(F)(F)C(CNC(=O)C(C)NC=O)C1 C#CCC(C)(C(=O)N1CCC(C)(N(C)C)CC1)NC(c1ccc(C)s1)=O C#CCC(CC(=O)N(C)CC1(O)CCC1)NC(=O)C(C)(O)C1CC1 C(CN=c1[nH]c(Cl)ncc1C)(CC(C)C)NC(c1c(CCC)cccc1)=O N1(C(C(C)(C2CC2)OC)=O)CC(CNC(=O)C2CC2)CC(C)(C)C1 c1(CC(=O)NCCOCC(=O)NCC2C3CCCC23)ccc(Cl)nc1 C1(CC=C)(NC(=O)C2=CCC2)CCN(C(C2CCC=CO2)=O)C1 c1(C(=O)NCC2N(C(CC(CC)C)=O)CC(O)C2O)nc[nH]c2ncnc1-2 C1(C#CC(=O)NC2(CNC(=O)CC3C=CCC3)CCCC2)(CC)COC1 C1(C)(CNC(C(C)O)=O)CCCN(C(=O)CCS(=O)(=O)N2CCOCC2)C1 CC(C)C(C)CS(=O)(=O)N1CCC(c2cccc(F)c2)CC1 N1(C=O)CCN(CC(=O)N)CC1.Cc1nonc1C1(NCCS(C)(=O)=O)CCC1 c1(OC)c(Cl)nc[nH]c1=NCC1C2CN(C(C3COCCO3)=O)CC12 C1(CC)C(C(=O)N(C)CCOC(F)F)CCN1C(c1oc(C)cc1C)=O CCCCC(C(=O)NC)NC(=O)C(CC)NC(=O)CN(C1CCC1)C C(=O)(C1=CCCC1C)NC1CC(CCNC(c2c(C)nc(CC(C)C)s2)=O)C1 C1(C(C(=O)NC(C(=O)NCCC(C)N(C)C)c2cccs2)=O)CCCCC1 C(=O)(CCCCC1CC1)NCC(CO)NC(c1cn(C)nc1)=O CC(C)(CN=c1nc2scnc2c(NCc2nc3ccccc3o2)[nH]1)CS(C)(=O)=O C(CC(O)CNC(=O)CCOCC1CC1)NC(=O)CO c1(SCCCCNC(C(C)n2cccn2)=O)cccc(OCC(=O)OCC#N)c1 c1(C(N2CC(NC(CC(C(=O)OC)(C)C)=O)C3C2C3)=O)cc2cccc(C)n2n1 C1(C(=O)NC(C)CCNC(=O)CC2(C#N)CCC2)(OC)CCCC1 N1(C(c2ccc(C(CC(C)C#N)C)cc2)=O)CCOC2(CC(O)C2)C1 N1(C(C(n2c(C)ncc2)C)=O)CC(NC(=O)CN2CC(CF)C2)CCC(O)C1 c1(CC(=O)N(C(C)CNC(c2c[nH]nc2OC)=O)CC)c(C)nn(C)c1Cl Cc1n[nH]c(C)c1CCC(=O)NC1CC1NC(=O)CCn1ncn(C)c1=O C1(OC)CC(CC(=O)NCc2cc(C3CC3)on2)N(C(=O)C=C(C)C)C1 n1(CC=C)nnnc1C(c1sccc1Cl)NC(c1cncs1)C C(=O)(C1=CCC(C)CC1)NCCC(C)NC(C(c1nccc(C)c1)(C)C)=O CCCC(CCCNc1nccc(CC(=O)Nc2cc(C)nc(C)n2)n1)OC.C(C)(C)C C1(C(N2CCC(NC(c3cscc3Br)=O)C2)=O)CCCCCCC1 Cc1ccc2c(c1)CC(C(=O)NC(C)CNC(c1sccc1Br)=O)S2 C1(OC)CN(C(C2CC2CC(C)C)=O)CCC1NC(c1cccc(Cl)c1F)=O N1(C(C(CC)COC)=O)CCC(CNC(=O)CC2(COC)CC2)C1(C)C c1(CCC(=O)OC(CC#CC)C(=O)OCC)c(C)nc2cc(O)nn2c1C c1(C(N(CC(C)NC(=O)C(C)(C)n2ccnn2)C)=O)nccnc1N C(=O)(CC(C)C(=O)NCC1CCC(C(=O)Nc2ccc([N+](=O)[O-])o2)CC1)OC CCC(CCOC)C(=O)NC(C1CC(NC(C2(C(C)(F)F)CC2)=O)C1)C c1(SC)nc(N2CC(NC(c3ccnc(C4CC4)c3)=O)CC2C)ncc1C CCCC(C)C(=O)NCCC1CSCCN1C(=O)Cc1conc1C c1(C(N(C2(C(=O)NCCc3cccs3)CCSC2)C)=O)sccc1C#N C1(COC)CCN(C(c2ccc(Cl)c(F)c2)C(=O)NCc2ccco2)CCO1 c1(C(C(=O)NC(C)(C)C)N(C(C(=O)OC)C)C)occc1Br C1(NC(C(C)(C)OC)=O)CCN(C(=O)C(F)C(F)(F)F)CCC1c1ccccc1 c1(C(N(CCCNC(CC2CC(=O)C2)=O)C2CC2)=O)ccc(OC(F)F)cc1 c1(N2CC=C(CCOC)CC2)nc2cccc(F)c2c(=NCCCF)[nH]1 C1(C(N(CC(O)C(C)(C)C)C)=O)CCN(C(c2ccc(N)cn2)=O)CC1 c1(C(=O)NC(CCNC(COCCOC)=O)C)cc2c(cc1Cl)OCCO2 N1(C(C(CCCC)O)=O)CC2CC(C1)N(C(=O)Cc1ccc3nn[nH]c3c1)C2 n1(C(C)C(=O)NC2CCN(CC=CCC3CCCCS3)C2)cnc2ccccc12 N1(CC(C23C(C)(C)C(CC2)CC3)=O)CCN2CCNCC2C1 CC1CCN(C(=O)C=CC(=O)NCC2CC2)C1CNC(=O)C(=O)NC1CC1 c1(C(N2C(C)(C(N3C(C)(COC)CC3)=O)C=CC2)=O)ccc(C)c(C)n1 c1(C(N2CCC(C)(NC(C3C=C(C)CS3)=O)CC2)=O)ccc(C#N)cc1F C(=O)(C(C)CC(=O)NCC=CCNC(c1nccnc1N)=O)OC N1(C(C)=O)CSCC1C(=O)NC(C)(C)C(C)NC(=O)C(c1ccc(Cl)s1)C CCC(CC(=O)NCC1CC(NC(=O)CC2CCS(=O)(=O)C2)C1)C(C)C N1(C(c2ccc(Cl)s2)=O)CC2CCCC2(C(=O)NC2C3CCCC23)C1 CC(C)(C)CC(O)CNC(=O)CCN(C(=O)C1=CCOCC1)CCO N1(C(c2n(C)ccc2)=O)CCCC(C)(C(=O)NCCc2ccc(F)nc2)C1 N1(C(c2c(C(C)C)con2)=O)CC2CC(c3ccccc3)C(C2)C1 C1(C(N2CCC(C(N(CC=C)CCOC)=O)C2)=O)CC(=O)N(C)C1 c1(C(N2CCC(NC(c3n(C)cnc3)=O)C23CCC3)=O)sc2ncccc2c1N Cc1ccc(-n2cc(C(=O)N(C)Cc3cc(Cl)ccc3F)nn2)cc1Cl c1(NC(C(CC)(C)CNC(=O)CCc2cscn2)=O)cnc2ncnn2c1 CN(C(=NCCN1CCOC(C)C1)NC1CCC(C)(C)C1)Cc1ccnn1C C1(O)(C(C)NC(C2C(CC)CCCC2)=O)CCN(c2cc(Cl)c(O)nn2)CC1 c1(C(N2C(C(N3C(C)(CC)CC3)=O)CCC2C(C)C)=O)ncnc(O)c1F N1(C(CCCCC)=O)CC2(CNC(=O)CCOCCOCCCO)CC(F)(C1)C2 N1(C(C(CC)N(C)C)=O)CCC(NC(C2CCC(C)C2)=O)CC1 C1(C(=O)NCC(C(C)C)NC(c2cn(C)nn2)=O)COc2ccc(Br)cc2C1 C1(CNC(C2CC3(CCO2)CC3)=O)CN(C(c2cccc(O)n2)=O)CCCO1 c1(C(=O)NC2C(NC(=O)CN3CC=CC3)CCOC2)ccc2ccccc2n1 c1(C(=O)NCC2CCC(NC(c3c(C)noc3C)=O)CC2)cccc(F)c1Cl C(CN=c1[nH]c(C)cc(=NC2CCN(C)C(C)C2)[nH]1)=C(C)CN1CCOCC1 c1(C(=O)NC2COCCN(C(C=CC)=O)C2)ccc2c(c1)N(C)CCO2 C#Cc1ccc(C(=O)NC2CC=C(C(=O)NC(c3ncc[nH]3)C)C2)cc1 c1(CCC)ccc(C(=O)NC2(CCNC(=O)CC3CCOC3(C)C)CC2)cc1 C(CC(C)(C)C)(C(=O)NCC1CC12CC2(F)F)NC(c1nn(C)c(C#N)c1)=O C1(C(=O)NCC(CC)NC(=O)C(C)OC(C)=O)(OC2CCOC2)CCCC1 N1(C(c2c(C)n[nH]c2C)=O)CC(C(=O)NCC=C2CCSCC2)CC12CCC2 C(=O)(C1=CCCCC1C)NC(C(=O)NCC1(C)CCC(C)CC1)CO N1(CCNC(C=CCN(C)CC)=O)CCCN(C(=O)C(F)C(C)C)CC1 C1(C)(CC)CN(C(c2c[nH]nc2CCNC(C2COC(=O)C2)=O)=O)CCO1 c1(C(=O)OC)ccc(O)nc1N1CC=CC(NC(=O)Cc2nnc(C)o2)C1 c1(C(=O)NC(CCOCC)C)cnc(CNC(=O)C(C(C)O)N(C)C)nc1 C(=O)(CCC(CF)CF)N1C(C(=O)NCCCCCC)CC(CC)CC1 C1(CNC(C(C)(C)c2cscn2)=O)CC2(CCN(C(=O)C(F)(F)CO)C2)CO1 CC1CCC(CNC(C2CCC(NC(C)(C)C)C2)=O)CC1 CC(C)C(C)CC(=O)N(C1CCCC(NC(c2ccnc(F)c2O)=O)C1)C n1(CCCOC)nc(C(=O)NC2CC(C)N(C(=O)C#CC(C)(C)C)C2)ccc1=O C1(CNC(Cc2cc(OC)no2)=O)CN(C(C2(C)CCCCO2)=O)CC1(C)C C1(O)(CNC(C2(OC)CCCC2)=O)CCN(C(=O)C(C)(C)n2cnc(C)c2)CC1 C(C)(CC1CCC1)(C(=O)NCCN(C1CCC1)C(c1cccc(F)c1)=O)NC(C)=O c1(OC)ccc([N+](=O)[O-])c(NC2CN(C(=O)C(C)=C3CCC3)C2)c1F c1(C(N2CCC(C(C)NC(c3c(CC)cccc3)=O)C2)=O)ccc2nnnn2c1 c1(NCCC(C=C)C)[nH]c(=NCCCCN)nc2c1ncn2C.SC Cc1occc1CC(N1C(CNC(=O)C(C)c2ccsc2)CC1C)=O c1(C(=O)NCC(N(C(CCCSC)=O)C)C2CC2)cnc(SC)n1C CCCCC(C)C(=O)NCCCCNC(=O)C1=CCCCC1 C1(NC(C2CC(OC(F)F)C2)=O)CC(CO)N(C(=O)CCN2CCCC2=O)C1 N#Cc1ccc(C(N2CCC(n3cc(C4CCCC(O)C4)nn3)C2)=O)[nH]1 C(CN=c1cc(C(N)=O)nc[nH]1)N1CCN(C(C2C(C)OCC2)=O)CC1 c1(C(N2C(C(N3CCCC(OC(C)C)C3)=O)COCC2)=O)ccnc(Br)c1Cl c1(CC)[nH]c(=N)sc1C(=O)NC1CCCN(C(=O)C=CCOC(C)(C)C)C1 C(=O)(CCC(F)(F)C(F)F)NC1C(NC(CCCC(=C)C)=O)C2CCC1C2 C1(CC(N2C(C)(C(=O)NCC3(OC)CCCC3)CC2)=O)CC2CCC1C2 c1(CC)cc([N+](=O)[O-])ccc1N1CC2CC(NC(C3C4COCC34)=O)CC1C2 N1(C(CC)=O)CCCC(C2CCCCN2C(=O)CC(=O)NCC)C1 N1(C(CSc2ccnc(OC)n2)=O)CCC(C(=O)N(CC(F)(F)F)CC)C12CCC2 N1(CCC(=O)N(CC(=O)Nc2c(C)nc(C)s2)C)C(=O)C2C3C=CC(C3)C2C1=O c1(C(C(C)C)NCC(=O)N(C2CCOC(C)C2)CCC)cc2ccccc2o1 c1(C(=O)NCC(C2CCN(C(C3CC34CC4)=O)CC2)(C)C)cc2n(c1)CCSC2 c1(NC)c(C(=O)NC2CCCCN(C(=O)C3=CCCO3)C2)cccc1N c1(C(=O)OC)cccc(SC)c1[N+](=O)[O-].C12CN(CCN(CC3CC3F)C1)C2=O N1(c2cc(OC)ncn2)CCC2(CCCN(C(=O)C3=C(SC)CCCC3)C2)C1 C1(C(=O)NCC(CO)SC2CN(C(N)=O)C2)(OC(C)=O)CCCOC1 C1(C(=O)OC)CCCCC1C(=O)ON1CCC(n2ccnc2)CC1 N1(C(C2CCN(C(=O)OCC)C2)=O)CCC2(CC2NC(=O)Cc2nonc2C)C1 n1(CC)c(=O)c(C)nc2cc(NC(=O)NC(C(C)(C)C)c3cccs3)ccc12 C1(NC(C(CC)(C)F)=O)CCC2(CC1)CC(NC(c1cccc(N(C)C)n1)=O)C2 c1(C(=O)NC(CC(C)NC(C=C(CC)CC)=O)C)[nH]c(=N)ccc1C C1(NC(C(c2ccccc2)OC)=O)CC(C)CN(C(c2cnc(F)c(Cl)c2)=O)C1 C1(NC(C(COC)C)=O)CN(C(=O)C(C)(C)CO)CC1(C)C N1(C(CCNC(C2CCN(CC)C2)=O)=O)CCN(C)C(=O)C1CC c1(C(N(CC(O)CNC(C2COC(=O)C2)=O)C)=O)c(-c2ccccc2)nsc1N Cc1ncc(CC(=O)NCC2(F)CC(NC(=O)CNC(c3ccco3)=O)C2)[nH]1 c1(C(=O)NCc2occ(NC(c3ccn(CCCC)n3)=O)n2)nc(C)nn1C N1(C(C(=O)NC2CCOC2)c2ccoc2)CCOCC1CCC#N C1(CC(=O)NCCCC2CC3CCC2O3)CCCCN1C(C1(CO)CC=CC1)=O C12(C(N(CCS(C)(=O)=O)C)=O)CCC(NC(=O)CC3CCC3)(CC1)C2 C(=O)(C(O)CCS(C)=O)NCCOC(c1nc(CC)n(C)n1)=O.C(C)(C)(C)O c1(C(=O)OC(CCCC2(NC(=O)OC(C)(C)C)CCC2)=O)cnc(C(C)(F)F)s1 c1(C(N(CC(CC)NC(=O)CC2CC(F)(F)C2)C)=O)cc2ccccc2c(=O)o1 C1(NC(=O)Cc2cnc[nH]2)CCOCC1NC(C1(c2cccs2)CC1)=O C(=O)(C(C)(C)CC(C)(C)C)N1C(CNC(C(CCC=C)(C)C)=O)CC(O)C1 N1(C(CCCC(C)=O)=O)CCCC2C1CCN2C(c1cc(F)cnc1O)=O C(=O)(CCC(=O)N(CC(O)CN(C)C(C1CC(CCO)C1)=O)C)N(C)C c1(C(=O)NCC2CCCN(C(C3C(CC)C3)=O)CC2)cc(=O)n(C)cc1Br Cn1cc(N(CC(N2CCCC2)=O)C(c2cc(CCN)on2)=O)cn1 N1(C(CC(CC)C)=O)CCN(C(C2(C3CC3)CC2)=O)CC1CF c1(-c2c(C)n[nH]c2)ccc(F)c(C(=O)NCC(C)N(C(=O)CC(C)C2CC2)C)c1 C1(CC(=O)NCc2ccncc2)CCCC(NC(=O)COc2ccon2)C1 c1(C(=O)NCC2CN(C(CCC(=O)NCCC)=O)CC2O)onc2ccccc12 C1(CN2C(CNc3ccnn3CC3CC3)CCCC2)CCc2ccccc2O1 CCC(O)C(C)(C)C(=O)NCCC(C)(C)NC(c1cccc(OC)c1N)=O C(=O)(C(C)(C)CCS(C)(=O)=O)N(CCN(C(C1CCn2c(C)cnc2C1)=O)C)CC C(CC(C)C)(C(=O)NC1CCCC1CC(=O)NCC1(CO)CCOC1)OC c1(CC)ccc(NC(=O)C=CC(C)NC(=O)CC2(C3CC3)CC2)c(C)c1 C12(CNC(C(COC)N(C)C)=O)CC1CN(C(=O)C(C)(C)n1cnc(C)c1)C2 C1(CCNC(CNS(CC)(=O)=O)=O)CCCN(C(=O)C(C)OCC(F)(F)F)C1 Cc1c(F)ccc(F)c1CNC1CC(C(=O)Nc2ccc(I)cc2C(F)(F)F)C1 c1(C(=O)NCC2CN(C(C(=O)NCC)=O)C2)ccc(C)s1 c1(N2CCC3(N(C)CC3)CC2)nc(NCCOC(C)(C)C)c2ncn(C)c2n1 c1(C(=O)NCC(C)NC(c2c(C)nns2)=O)cc(C(F)(F)F)ccc1O N1(C(=O)NC(CC=C)CC)Cc2ccccc2C12CCOCC2 C(=O)(C(C)C=C=C)N(C(C(=O)N(C(C=C)C1CC1)C)(C)C1CC1)C CC1CN2CCN1C(C(N1CCC(NC(C3CC(C)N(C)C3)=O)C1)=O)C2 C(=O)(C(F)(F)C(F)F)N1CCCC(N2CCN(C(CCNC(=O)CO)=O)CC2)C1 N1(C(c2noc(C)c2C)=O)CC(NC(c2cc(=O)ccn2C)=O)CC(C)C1 C1(CC)OCCC1C(=O)N(CCCOCCN(C)Cc1c[nH]nc1C1CC1)C CC1SCCCC1C(=O)NC(CN(C)C)C(=O)Nc1cnc(C(C)C)nc1 c1(CCOCC)cn(C2CCC(C(=O)NCc3nc(-c4ccsc4)no3)C2)nn1 C1(C(=O)NCCC(O)C2CCCC2)COCCN(C(c2cc(Cl)ns2)=O)C1 C(C(CC(C)C)C(=O)N1CCC(C(=O)NC)C1)NC(C1(CC)CC1)=O C1(NC(C=CC=CC)=O)CN(C(c2sncc2CC)=O)C2CCCC12 CC1CN(C(=O)CC2(CO)CC2)C1C(N1CCC(c2ncco2)C1)=O c1(C(N2C(CNC(c3n(C=C)ncc3)=O)C(C)CC2)=O)nc(SCC)ncc1Cl Cn1c(C(=O)NC2(CO)CCCN(C(C3CSC3)=O)C2)cc2sccc12 C(=O)(CC(C(C)C)C(C)C)NCC1(F)CCN(C(c2c(OC)csc2)=O)C1 C#CCC(C(=O)NCc1ccc(C(N)=O)o1)NC(=O)C(C)CCN(C)C C(N=c1nc2c(ncn2C)c(NCC2(CC)CC2)[nH]1)c1cnc(CC)s1 c1(OCC)nc(Cl)ccc1C(=O)NCC1CC2CCC1N2C(=O)C1=COCCC1 C(C(C)C(=O)NCC1(CNC(=O)C(F)OC(F)(F)F)CCCC1)SC Cc1cc(C(=O)NCC(C)NC(c2c[nH]nc2-c2ccccc2C)=O)ncc1F c1(CCC)cc(C(N2CCC(CNC(c3cc(=O)n(C)cn3)=O)C2)=O)cc(O)n1 C1(C(=O)OCC)CCCCN(C(C2CC3CCC2N3C(c2nocc2C)=O)=O)C1 C1(N(C(CCC)=O)CC)CCCN(C(=O)CC2CCCC23CC3)C1 C(=O)(C(C)(CCO)N(C)CC)N1CC(C(C)NC(=O)OCC)C1.C(C)(C)(C)OC(C)=O CCC(F)(F)CC(=O)NCc1cc(O)nc(CNC(c2scnc2C)=O)n1 C(=O)(CC(C)(C)NC(C1(C)CCCO1)=O)N(C(CC#CC)C)C c1(C(=O)NC2C(CNC(C(C)OCC)=O)CC2)ccn(C)c(=O)c1 c1(CC2(NC3(c4n(CCC)nnn4)CC4CCC3C4)CC2)ccc(Cl)c(COC)c1 N1(c2snc(C)n2)CC2CC1CCC2NC(C1CCc2nn[nH]c2C1)=O N1(C(c2ccc(SC)cc2)=O)CC(CNC(c2ccco2)=O)CCC1C c1(NC(c2cnccc2C(F)(F)F)=O)cc(-c2ccc(CO)s2)ccn1 CC(C(=O)NCC(C1CCCC1)NC(=O)C(=O)NCC(F)F)C(C)(C)C c1(C(N2CCC(CN(C(CN(C(=O)OC)C)=O)C)C2)=O)ccnc(S(N)(=O)=O)c1 CCC(CC(=O)NC(C)C(CO)NC(C1CC(F)C(=O)N1)=O)C(C)C Cc1cc(NC(c2cc(N(C)C)cc(Br)c2)=O)ncc1F.C12(F)CCCN(C1)C2 Cc1cc(C(=O)NCC2(F)CCC(NC(C3(C)CC3(Cl)Cl)=O)C2)ncn1 Cc1nn(C)c(NC(C2CN(Cc3cscc3Br)CCO2)=O)c1Cl Cc1cc(Cl)ccc1C(=O)NC(CNC(=O)Cc1cncnc1)C1CC1 CC(CC(N)=O)C(=O)NCc1ccnc(C(=O)NC(C)(C)C(N)=O)c1 C1(C(=O)NCC=CCSC)CCCN1NC(=O)CCOCC1CC1 c1(C(N2C3CN(C(C(=O)NCC)=O)C(C3)C2)=O)cccc2c1CC(C)(C)C2 CC(C)(CNC(=O)COC1CCCC1)CC(=O)NC1(C)CC1(C)C C1(NC(=O)NCc2cn(CC)nc2)CC2CCC1N(C(=O)OC(C)(C)C)C2.OCC c1(OC)cc(C(N2CCC2CNC(C2(CCF)CC2)=O)=O)cc(N)c1N C1(NC(CCc2ccn(C)n2)=O)CN(C(=O)C=Cc2ccccc2)CC2(CC2)C1 S(=O)(=O)(c1cccc(CNC(=O)Nc2cnc3ccc(F)cn23)c1)N(C)C c1(NC(C)=O)cccc(C(N2CC(NC(=O)CCOCC3CC3)CC2C)=O)c1C C1(C(=O)NC2CC(NC(C3CC4OC(=O)OC4C3)=O)C2)Cc2ccccc2O1 c1(CCC(=O)NC(CNC(CC(C=C)C)=O)C2CC2)cccc2c1OCCO2 n1(CCC(=O)NC(CC(C)NC(C=C(C)C)=O)C)cnc2cc(F)c(F)cc12 Cc1nn2ccccc2c1C(=O)NC(CO)C(C)NC(=O)C(c1ccnn1C)C N1(C(=O)COCC2CCOC2)CCN(C(c2coc(C(F)F)n2)=O)C(C(F)F)C1 N1(C(c2c(OC)ccnc2)=O)CCC(C(F)(F)F)C(NC(=O)CCN2CCC2)C1 C1(NC(CCNC(C(C)(C)C)=O)=O)CC2(C1)CC2C(=O)NC1C2CCC1CC2 C(=O)(C(CC1CC1)NC(=O)CCn1cccn1)N(C1CC(OCC)C1)C C1(O)(C(=O)NCC2C(CC(=O)NCc3cccnn3)C2)CCCCC1 C(=O)(C(F)CC(C)(C)C)NC1CCC(CC(=O)NC(c2n(CC)ncc2)C)C1 N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2NC(C1(F)CC=CCC1)=O O=NN1CCCCC1C(N1CCC(F)(CNC(=O)CC2CC3CCC2O3)C1)=O c1(C(=O)NC(C2CCN(C(C(C)NC(=O)OC)=O)CC2)C)ccc2nncn2c1 C1(C(S(=O)(=O)C(C2CCC(C)(C)CC2)C)C)CCC(F)(F)CC1 C(=O)(CC(C)C(C)(C)NC(=O)Cc1cnsc1)N1CCC(CC(C)C)CC1 N1(C(c2c(C)cnnc2)=O)CC(CO)C2(C1)CN(C(C1(F)CC=CCC1)=O)C2 N1(C(Cc2nc(C)sc2Cl)=O)CC(NC(=O)C(N2CCNC2=O)C)CC(F)C1 C1(NC(CC(C)C2CC2)=O)CCSC12CN(C(c1cnc(N)cn1)=O)C2 C1(CNC(CC(=O)NCC#C)=O)CC2CCC(C1)N2C(=O)C(C)CC(C)C Cc1no[nH]c1=NC(=O)c1n[nH]cc1NC(c1ccc(Cl)c(Cl)c1Br)=O C(CC(CC)C(=O)N(CC(C)CCC)C(C(=O)CC=CCC(=O)NC)CC)=CC C12(CC#C)CCN(C1)CC1CCN(C1)C2=O.c1(C(=O)OC)ccc(OC)nc1 n1(CC(=O)NC(CNC(C2(F)CC=CC2)=O)C2CC2)nnn(-c2cccs2)c1=O C(c1cc(Cl)ccc1OC)=C(CN1C2CN(C(C(CCC#C)O)=O)C(C2)C1)C CCC(C)(CNC(=O)CSCCC#N)NC(C1CC1c1ccc(Cl)s1)=O C(C)(C(=O)N1CCC(NC(C2(CCF)CCOCC2)=O)C1)(C(C)C)NC(C)=O C1(C(=O)NC(c2cccc(F)c2)C)CCN(C(c2ncnn2C)=O)CC1O c1(C(c2nnnn2C2CCC2)NC(C(C)C)C2CCC2)c(Br)n[nH]c1Br c1(OC)cc(-c2cn(CCCC(=O)NCCOC)nn2)ccc1Cl CS(=O)(=O)c1cc(C(=O)NC2CN(C(C3(CO)CC3)=O)CC2O)co1 C1(C(C(C)NCCC(c2cccc(F)c2)O)OC)CCC(F)(F)CC1 c1(C(=O)NCCCN(C(c2cnc(=N)[nH]c2)=O)CC)ccc2c(n1)CCCC2 N1(C(C2CC(C#C)(O)C2)=O)CC2CCC(CNC(=O)CC(CC)C(F)F)C2C1 CN(C1CCc2cc(Cl)ccc21)C1CN(C(=O)CN2CCCC2)C1 C1(NC(CSCCOC)=O)CN(C(=O)CN2CCOCC2=O)CCC1C(F)(F)F C(=O)(CC1=NNC(=O)C1)N1CC(F)(CNC(C(C)N(CC(F)(F)F)C)=O)C1 C1(C(N(C)CC2(O)CN(C(C(C)Sc3cccs3)=O)C2)=O)C2CC3C(C2=O)C13 C1(NC(C(C)SC)=O)CN(C(=O)Cn2ncn(C)c2=O)C2CCCCC12 CC1(C=CCO)COC1.CC(CCNC(=O)COCC(F)F)OC C1(C(N2C(C(=O)OC)C=CC2)=O)C=CCN(C(=O)C(CC2CC2)OC)C1 CCCS(=O)(=O)CC(=O)N1CCCC(COC)(NC(=O)C(C2CCOCC2)F)C1 c1(-c2c(OCC)cc(Cl)cc2)n[nH]c2c1CN(C(c1cc(COC)[nH]n1)=O)C2 CC(CN(C)C)CC(=O)N1CCCC(CN(C)C(c2cn(C)nc2O)=O)C1 S(=O)(=O)(c1ccc2oc(=O)ccc2c1)N1CC2N(C(c3cc(Br)cc(Br)c3)=O)C2C1 CC1CC(NC(=O)CC(C)(C)c2ccccc2)CN(C(=O)CCc2ccc[nH]2)C1 N(C(=NCCOCCN(S(C)(=O)=O)C)N1CCC(C)(C)C1)Cc1c(F)ccc(C)c1 CCC(CC(F)(F)F)NC(C1CC(CNC(=O)C=Cc2ccc(C)o2)C1)=O N1(C(c2cnc(CC(C)C)s2)=O)CC(CNC(=O)CC2(C(F)F)CC2)C(C)(C)C1 C1(C(N2CC(C#CC)C2)=O)CN(C(=O)COC2CCC2)C(C)(C)C1 c1(C(=O)NC(C(C)C)CNC(=O)COCC2CC2)cc2cccnc2[nH]1 C1(C(=O)O)(NC(C(=O)OCC)CO)Cc2cc(Cl)ccc2C1 C1(C(N2CC3(CCN(C(C(C(C)C)(C)O)=O)C3)C2)=O)CC2CC(O)CC(C1)C2 C1(NC(c2c(C)cc(O)cc2C)=O)CS(=O)(=O)C2CN(C(=O)CCCCF)CC12 c1(N(C)CCNCCCC)ccc(S(=O)(=O)N(C)CCc2ccccn2)c(Br)c1 CC(C)(C)C(=O)CCC(=O)N1CC=C(C(N2CC3CCCCC3C2C)=O)C1 C1(CCC(C)C)CCCCN1C(=O)NC(C)C(C)(C)C(=O)OC(C)(C)C C1(C(=O)NC(CNC(c2c(C)nsc2)=O)C(C)C)CCCN1C=O c1(N2CCC(NC(C(CC)C)=O)C2)ccccc1OC(c1ccccc1)C#N CCC(CCC(=O)N1CC2CC1CN2C(c1cccnc1O)=O)OC CCC(CSC)(c1nnnn1CC(F)F)NCCOC1CCCC1O c1(C(N(c2nccc(OC)n2)C)=O)ccc(C)c(C)c1.C12CCC(C1)N2 c1(C(=O)NCC2CN(C(COCCCCC)=O)C2)c(Br)c(C)nn1C c1(C(=O)NCC2N(C(c3cc(C#N)no3)=O)CC2)ccc(S(=O)(=O)C2CC2)cc1 C1(NC(C2(OC)CCSC2)=O)CCN(C(c2ccccc2SC)=O)CC1C CC1=C(C)CC(C(=O)NC2CC3(C2)CN(C(=O)COC2CCOCC2)C3)CC1 O=C1Cc2cc(C(N3CCc4ccccc4C3)=O)ccc2CN1 C(=O)(C(C(C)NC(=O)CCC1CC1(F)F)C(C)C)N(CCOCC=C)C C1(CNC(=O)NCCN2CC3CC(C2)O3)CCCCN1CC12CCC(CO1)C2 c1(CCN=C(NCc2scc(CC)n2)NCC2CCSC2)ccc2occc2c1 Cc1cc(C(=O)NC2CCN(C(=O)CN3CC=CC3)CC2C)cc(C)c1Cl c1(OC)cc(C(=O)N(C(C)CN(C)C(C2CCC(CO)CC2)=O)C)c(O)c(Cl)c1 c1(OC)ccc2c(c1)NC(=O)C2CC(=O)NCc1nncn1C(C)C Cc1cc(C)n(CC2(C(N3CCC(OC4CN(C(=O)C(N)=O)C4)CC3)=O)CC2)n1 N1(C(c2cn(CCCC)nn2)=O)CCN(C(c2nn(C)cc2C)=O)CC1CC c1(OCC)ccccc1C(=O)N(CCC(=O)NC(C(N)=O)C1CC1)C Cc1sc(C)cc1C(=O)NCC1CC1C(=O)NC(C)CC(C)O N1(C(c2c(CC=C)cccc2)=O)CCC2C(NC(=O)CC3(C)CC(F)(F)C3)CC12 Nc1cc(O)cc(C(N2CCC(n3cnc(C(F)(F)F)n3)C2)=O)c1Br c1(C(C)=O)ccc(C(=O)NCCCN(C)C(c2ccc(OCF)cc2)=O)c(Br)c1 C1(C(=O)NC(c2ccc(OC(F)F)cc2)C)CCC2(CCC1(F)F)OCCO2 Nc1cccn(CC(N2CCCC(CNC(=O)CCC3CCCC3)C2)=O)c1=O CON=Cc1ccc(C(=O)NC2CCN(C(C3(OC)CCC3)=O)CC2CO)cc1 c1(OC)ccc(C(=O)NC2C3CC2N(C(=O)C(c2cncnc2)C)C3)nc1 c1(C(N2CC(NC(COc3cc(C)on3)=O)(COC)C2)=O)nnn2c1CCCC2 CN1CCCC(CNC(C2CCCN(C(c3csnc3Cl)=O)C2)=O)C1 C1(C(N)=O)CCC(C(N2CC(N3CCN(C(C4CCCO4)=O)CC3)C2)=O)CC1 C1(O)(CN(C(c2c(OC)nsc2)=O)C)CCN(C(C2CCCN2C(C)=O)=O)CC1 c1(OCC)ccc(C(=O)NC2CCC(CCC(C)C)C2)cc1Cl c1(CC)cccc(C(=O)NC2CCCC2C(=O)NCCCCNC(N)=O)n1 C(CC(=O)N1CCS(=N)(=O)CC1)(C(F)F)NC(c1n(C)ccn1)=O N1(C(c2cncc(F)c2)=O)CC2CCC1C1CN(C(C3C=CCCC3)=O)CC21 c1(C(C(N2CCCC(CNC(C3(CO)CCCC3)=O)C2)=O)O)ccccc1F c1(OCCC)ccc(C(=O)NCC2COC(CNC(=O)Cn3cncn3)C2)cc1 CON(CCC(=O)N(C1CCC1)C1CC1)C(=O)CC(C)C(F)(F)F CCCCC(CC)CC(CNC(=O)Cc1nc(C2CC2)n[nH]1)CC N1(C2CCN(C(C3CCOCC3)=O)C2)CCN(C(C2(C)CC2Br)=O)CC1 N1(C(CCC(=O)OC)=O)C2CCCC1CC(NC(=O)Cc1ccc(F)c(Br)c1)C2 Cc1ccc(C2CC2C(=O)NC2CN(C(=O)CC3CC=CCN3C)CC2O)cc1 C1(CNC(CSCCN(CC)CC)=O)CC(C)N(C(=O)CC2CCCO2)C(C)C1 c1(C(=O)OCC)cnc(NC(C2CC(O)CN2C(c2cncnc2)=O)=O)nc1 n1(C2(NC)CC2)cccn1.C1C(=O)NCCC2(CC2)C(=O)N1C.CC CCC(C)(C)C(O)C(=O)N1CCC2(NC(c3nc(O)sc3C)=O)CCCC12 CCC(C(=O)NCC1CN(C(c2cnc(C3CC3)nc2C)=O)C1)C(C)(F)F c1(C(=O)NC2(COC)CCN(C(c3ccsc3C)=O)C2)[nH]nc2c1CCC2(C)C C1(C(=O)OCC)CC2COCC(C1)C2NC(c1cnc(COC)o1)=O C1(NC(c2c(C)cc(C)s2)=O)(CNC(C2CCCC2)=O)CCCCC1C c1(CCC(=O)NC(C)CN(C)C(C2CCCO2)=O)cncc(F)c1 c1(C(N2CCCC(CCNC(c3c(CC)occ3)=O)C2)=O)sc(C)c(C)c1C CC1C(NC(c2cc3occc3[nH]2)=O)CCCN1C(=O)C=Cc1ccccc1 Cc1ccc(C)c(C(=O)N(CCCCN(C(=O)C(C)Cc2ccccn2)C)C)c1 CC1CCN(C(C2(c3cccs3)CC2)=O)C(CNC(=O)C(CCO)N(C)C)C1 N1(C(C(C(C)C)n2cccc2)=O)CC2(CCNC(C3(N(C)C)CC3)=O)CCC1CC2 CC(C)CC(CN=c1ncc2ccccc2[nH]1)NC1CCCCCC1 C1(NC(C(C=C)O)=O)CCN(C(c2[nH]cc3c2CCCC3)=O)CCC1(F)F C1(CC(=O)N(C)CCN2CCCC2=O)CC(O)CN1C(=O)C=Cc1ccn(C)c1 c1(NC(C(=O)NC(CC=C)Cc2ccccc2)=O)ccc(S(=O)(=O)C2CC2)cc1 c1(OC)ccc2c(CNC3CC4(C3)CC(C(=O)NCC(C)O)C4)c[nH]c2c1 C1(CCC(C)C)CCCN(C(C2CN3CCC2C3)=O)C1 CCC(C)C(C)CN=c1[nH]c(=NCc2ccccc2CO)[nH]c2cccc(F)c12 c1(C(=O)NCC2C(C)CN(C(=O)CC3CCS(=O)(=O)C3)C2)ccnc(Cl)c1F C#CC(CC)(CC)NC(=O)CC(CC)N(C(=O)C(C1CCCCC1)=O)C c1(C(=O)NCC(=O)NCC2(NC(C3(C4CC4)CC3)=O)CC2)cc(Cl)ccn1 C1(NC(C(c2ccccc2)C)=O)CCN(C(=O)C(C)n2ccnc2)C1(C)C C=CC(C)(CC)C(=O)N(CCC(=O)NC1CN(C)CC1OC)CC C(=O)(CC(C)(C)C(F)F)N(C1CCCN(C(c2ncsc2S(N)(=O)=O)=O)C1)C C1(C(=O)NC(c2ccn(C)n2)CC)(CC)CCCN1C(c1cnc[nH]c1=N)=O C1(CNC(C2(CC)CC2(F)F)=O)(CNC(=O)C=CC(=O)N(C)C)CC12CCC2 c1(OCC)cccnc1C(=O)NC1CCCC(CNC(c2cnc(S)nc2)=O)C1 n1(CCOC)cnnc1NC(C)C(=O)OCC(=O)OC(C)C CCC(C)CC(C)N(C)C(C1(NC(c2ccncc2F)=O)CSC1)=O c1(C(=O)NC2(C)CCCN(C(C(C(=C)Cl)(C)C)=O)C2)cnc2c(C)cccn12 C1(C)(CC)C=C(C(=O)NCC#CCNC(=O)CC(C)c2cccnc2)C1 CC1CCCCC1OCC(=O)NCCCN(C(=O)Cc1cnn(C(C)(C)C)c1)C N1(C(C2CC(F)CCN2C(C2CCC(C(N)=O)C2)=O)=O)CC(C2=NOCC2)C1 N1(C(c2c(OCC)cccc2)=O)CCN(C(=O)CC2CCCNC2=O)CC(O)C1 CC1CCCC1(O)Cn1cc(-c2ccc(N(C)C)cc2)nn1 NC(Cc1ccc(C(N2CCCC2Cc2ccncc2)=O)cc1)CC(F)F c1(CC(=O)NCC2C(NC(C3(C=C)CCC3)=O)C2)cc(Cl)ccc1Br CC(C(=O)N1CCN(C2CCC(NC(C3C4CNC(=O)C34)=O)C2)CC1)C(C)O C1(C(N(c2ccc([N+](=O)[O-])cc2)C)=O)C2CCCC2CN1C(=O)NC(C)(C)C Cn1ncc(Cl)c1C(=O)N(CC(=O)NCC(C)(F)F)C1CCC1 C1(C)(C(=O)NC2CCN(N3CCN(CC)CC3)C2)CCC(NC(=O)OC)C(C)C1 C(=O)(CC1=CCOCC1)N1CCC(NC(c2c(C)noc2)=O)C1CC(F)(F)F N1(C(c2c(C(C)C)con2)=O)CCN(C)C(C(=O)NC(C(F)(F)F)C2CC2)C1 c1(C(=O)NCC2(F)CCN(C(Cc3nc(C)sc3)=O)C2)ccc(OC(F)F)nc1Cl C1(CNC(C2(COC)CC2)=O)CN(C(c2csc(C)c2)=O)CC12CC2 N1(C(CC=C)=O)CCC(CCNC(=O)C=CCN(C)CC)(COC)CC1 Cc1ccc(C(F)(F)C(=O)N2CCC(CNC(C3C4CCN3CC4)=O)C2)cc1 S(=O)(=O)(c1cc(Cl)cc(Cl)c1O)NC1CN(Cc2ccc(C(N(C)C)=O)cc2)C1 Cc1cc(C(N2CCC(C)(NC(c3cnoc3C3CC3)=O)C2)=O)nn1C1CC1 C1(C)(c2cn(CC3CN(C(c4c(CC)ocn4)=O)C3)nn2)CCCN1C CC(C)C(CO)C(=O)N1CCOCC1CN(C(=O)C(F)(F)c1ccccc1)C Cc1cc(C(=O)NCCOCCn2cc(-c3cccs3)nn2)cnc1O N1(CC(=O)NCC2N(C(Cc3nc(CC)sc3)=O)CC2)C(=O)CCC1=O N1(CC)CCCC(C(N2CCC(CNC(c3c(N(C)C)c[nH]c3C)=O)C2)=O)C1 Cc1cc(C(N2CCC2CNC(c2ccc(CC#N)cc2)=O)=O)n2nccc2n1 N1(C(C(C2CCC2)OCC)=O)CCCCC(CNC(=O)CN(C2CCCC2)C)C1 C=CC1COCCN1C(=O)COC1CCN(C(C2CC3(CCO2)CC3)=O)C1 C(=O)(C(C)CC(=O)NCC1CCCC1C(=O)Nc1cnn(C2CC2)c1)OC c1(C(=O)NC(C(C)NC(c2ccc(CC)nc2)=O)C)ccc(C(C)C)cc1F c1(C(=O)NCC2(O)CCCN(C(=O)CC(F)F)C2)n[nH]c2c1CCOC2 Cc1c(C(=O)NC(C)CC(C)NC(c2ncc(F)cc2F)=O)nn(C)c1Br Cc1ccc(C(=O)NC2(C)CCN(CCCOC3CCCC3)CC2)c(F)c1F N1(C(CCCCC#C)=O)CCC(C2CC2)(CNC(=O)C(C)(C)C#N)C1 C1(CN(C(c2nc(Cl)sc2C)=O)CC)CCN(C(C2COC(C)C2)=O)CC1 c1(C2C(C(c3cccc(Cl)c3)Nc3c(C)nc[nH]3)CC2)ccc(Cl)cc1 c1(SCC)ccccc1C(=O)NC1CCC(NC(C2CC2OC)=O)C1 CCCCC(O)CC(=O)NC(C)(C)CCC(=O)N(CC(=O)OC)C1CC1 N1(C(c2ccncc2F)C(=O)NC)CC2CC(CF)C(C2)C1 N1(C(c2[nH]cc(CC)c2)=O)CC2CCOCC2(NC(c2cc(Cl)n(C)n2)=O)C1 c1(C(=O)NCC2(F)CCC(NC(COC(C)C)=O)C2)ccnc(F)c1F N1(C(c2ccc(OC(C)C)nc2)=O)CCC2C(C1)CN2C(=O)C(C)CN(C)C c1(C(=O)NC(CCCC)CNC(c2cnn[nH]2)=O)ccc(OC)cc1F N1(C(C2CN(C)C(=O)N2)=O)CCC(O)C(N(C(=O)CC2CCN(C)C2=O)C)C1 N1(C(Cc2c(C)non2)=O)CC(NC(c2cnnn2C2CC2)=O)CCC1C C1(NC(C=CCN(C(=O)CC2CCC(C#N)C2)C)=O)CCCC1C#N C1(NC(c2ccc(CCC)cc2)=O)C2CCC1N(C(C1CC13CCSCC3)=O)C2 C1(CNC(CSC)=O)CC2(CCOCC2)CN1C(=O)Cc1nocc1C(C)C Cc1ccc(O)cc1C(N1CC2CC(NC(=O)C(C)Cn3ccnc3)C1C2)=O c1(CCCN(C(=O)Cn2cc(CN3CCCC3)nn2)C)ccc(Cl)cc1 c1(C(C)C)ccccc1CS(C)(=O)=O.C12CC(C1)CN2C CC(C)C(O)CC(=O)NOC(CCc1ccc(F)cc1)C(=O)O N1(C(CNC(=O)C(Cl)Cl)=O)CCN2CCCCC2C1.O=C1CC=CCN1 c1(C(N2CC(C(C)C)C(NC(=O)CCC(C)(C)C)CC2)=O)nnn2ccccc12 N1(C(CN(c2ccccc2)CC)=O)CCN(C(C2CC2(F)Cl)=O)CC1 c1(C(=O)N(CCCO)Cc2ccn3nnnc3c2)cc2ccccc2o1 N1(C(c2c(C)nc(OC)s2)=O)CC2CCN(C(=O)C=CC(C)(C)C)C2C1C N1(C(CCOCC#C)=O)CCC(NC(=O)CC2CC(OC)C2)C(CO)CC1 c1(C(=O)NCC(C)NC(C2CC2C(C)(C)C)=O)ccc([N+](=O)[O-])n1C C1(C(=O)OC)CC(ON=C(C(=O)N(C2CCOCC2)CCC)C)C12CCC2 C1(C(N2CCC(OC)CC2)=O)COC2(CCN(C(c3cc(Cl)cc(Cl)c3)=O)CC2)C1 C(c1cc(Br)cs1)=CC(=O)NC(CN(C(C(=O)N(C(C)C)C)C)C)C c1(C(=O)NC(CC)(C)CNC(=O)C(C)NC(=O)COC)cc2ccccc2[nH]1 C(=O)(C1=CC2CCCCCC12)N1CCCCC(CNC(=O)NCCNC(OCC)=O)C1 C1(CC(=O)NCCC(C(C)C)NC(C2CCCC(C)C2)=O)CCC2(CCC2)O1 C1(CNC(CC(C)c2ccccc2)=O)(NC(=O)OC(C)(C)C)CCS(=O)(=O)C1 c1(COC)ccc(CCC(=O)NCc2cn(CCc3ccnn3C)nn2)cc1 C1(NC(C=CCC)=O)C=CC(CNC(C2CN(C3CCCCC3)C2)=O)C1 c1(OCC)ccc(C(=O)NC2CN(C(c3cc(OC)c(C)nn3)=O)C2)nc1OC c1(C(=O)NCC2CN(C(c3cccc(C(C)(F)F)c3)=O)C2)cc(F)c(O)c(Cl)c1 C1(C(=O)NCc2cccc(C)c2C)CCN(C(C2COCCC2C)=O)C12CCC2 CN1CCC(C)(C(=O)NCC2CCCCN2C(=O)COCC2CCOC2)C1=O c1(C(=O)NCC(CC)NC(c2[nH]c(O)nc2C)=O)c(-c2ccccc2)cn(C)c1C N1(C(C(CC)C2CCC2)=O)CCC(C)(C)C1CNC(=O)COc1cccc(C)c1 c1(CC)nnc(N2CCC(Oc3cccnc3)C2)n1CCCCOC C1(C(=O)NC2C(NC(=O)Cn3ncc(Br)n3)CCC2)CC2(CC2)CO1 N1(C(c2cc(C)no2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1CC1CC1 C1(N(C(c2c(C)nc(-c3cc[nH]n3)s2)=O)C)CCCN(C(C2CC2(F)F)=O)CC1 N12CC3CC(C3C1)NC(=O)CCOc1ccc(Cl)cc1CC2=O.CCCN.OC c1(C(N2CCC(C=CC(=O)NOC(C3CC3)C3CC3)CC2)=O)ncnc(O)c1F c1(NC(CSC)=O)ccccc1NCCN1CCCCCC1 c1(CC(=O)NC(CC)CNC(=O)CCCOc2cccnc2)cc(F)ccc1F c1(C(N2CC=CC(NC(C3CC34CC4)=O)C2)=O)ccc(C(F)(F)F)c(O)c1 c1(C(N(CC(C)OCC)C(C)C)=O)nc2n(c1Cl)CCCC2 N1(C(c2nc(C)n(C)n2)C(=O)NCCC#N)CCC(O)(CN(C)C)CC1 O=C(C(O)CC1CCCCC1)NC1CC(NC(c2snnc2C2CC2)=O)C1 n1(CC)ncc(C(=O)NCC2CCCC2NC(=O)C(n2ccc(C3CC3)n2)C)n1 C#CCC(C)(CC)C(=O)N1CCC(=CCNC(=O)C=C(CC)CC)CC1 C(C(CC(F)(F)F)NC(=O)CCCCF)NC(C(CC=C)C)=O c1(C(=O)NCCC2CCCN(C(C(CC)(C)CO)=O)C2)cc2n(n1)CCN(C)C2 c1(CC(=O)NC(c2nocc2C(N2C3CCC2CC3)=O)C)cccnc1O C1(CNC(c2c(COC)nn[nH]2)=O)C2CN(C(=O)C=CC(C)C)CC12 C1(C(=O)NCCCCCO)(CC)CCCN1C(c1ncccc1F)=O CCC(CC(=O)NC1CCCCC1NC(=O)CNC(=O)CC1CCCCC1)OC Nc1ccc(C(=O)NCC2(CNC(=O)C=Cc3ncc[nH]3)CCCC2)c(Cl)c1 c1(C(C(=O)NC(C(=O)NCCC(=O)OC)C)(F)F)cc(Cl)ccc1Cl c1(C(N2CC(c3ccsc3)OC(C)C2)C(=O)NC)cc(Cl)c(I)cc1Cl c12ccc(Cl)c(c1)C(=O)N2.C(C(=O)NC(CO)C(=O)OC)(C1(O)CCC1)OCC CC1(C)CC=C(C(=O)NC2CC(=O)N(C3CN(Cc4ccncc4)C3)C2)CC1 C1(CCC)CCC(c2cn(C(c3ccccc3)CC)nn2)CC1 c1(-n2cc(CCSCC)nn2)cccc(NC(=O)Cc2cccs2)c1 c1(COC)cccc(C(=O)NCC2CC2NC(c2n[nH]c(C3CC3)c2Cl)=O)c1 C(C(CC(F)(F)F)NC(c1ccc(=O)n(-c2ccccc2)n1)=O)NC(C(C)O)=O N1(C(CSC(C)=O)=O)CC2CCN(Cc3ccc(I)c(F)c3F)CC2C1 CCCCCCCCCC(=O)NCC1N(c2cc(O)ncn2)CCC1(C)C C(=O)(CCCCCN(C)C(c1nnn(C)c1N)=O)N(CC(CN(C)C)O)C N1(C(C=CC=CCC)=O)CCC(OCCCNC(=O)C2=CCSC2)CC1 C#Cc1cnc(C(=O)NCC2(F)CCN(C(C3COC(C)C3)=O)CC2)c(C)c1 C1(NC(=O)C=C2CCC2)(CF)CCN(C(=O)Cc2csc(-c3cccnc3)n2)C1 C1(O)(CNC(=O)CN2CCCCC2=O)CCCN(C(=O)Cc2cccs2)C1 c1(C(N(C2CCC(NC(CN3CCC(C)C3)=O)C2)C)=O)ccc2c(c1)COCC2 c1(C(=O)NC2CCCN(C(=O)CCCNC(N)=O)C2)ccn2ncnc2c1 C1(CN(CC)CC)CCCN(C(c2ncncc2OC)=O)CC1 N1(c2n(C)ncc2)N=C(C(=O)N2CCC(CO)=C(F)C2)CCC1=O.C1(=O)CO1 c1(C(CC)C)cc(C(=O)NC2CCC(NC(=O)Cn3nccn3)C2)on1 c1(C(=O)NC2(C)CC(NC(=O)C=C3CCC3)C2)cc(F)c(Br)cc1F c1(NC(C2CCCN(C3CCC(Cc4ccccc4)CC3)C2)=O)ccc(Br)cn1 c1(CC)nc(Cl)nc(N2CCC(NC(c3cc(C4CC4)on3)=O)C2)c1C#N C1(C(=O)NCC(C)(C)CCO)CCC(O)CN1C(=O)C=CC(F)(F)F C=CCC(CC(C)C)C(=O)NC(CNC(=O)Cn1cccnc1=O)CC(F)(F)F C(CC(C(=O)N1CC=CC(N(C)C)C1)NC(=O)Cn1cccnc1=O)OCC CCC(CC)CC(F)C(=O)NCC(C)C(F)C(=O)NC(c1ncc(C)[nH]1)CC C1(NC(Cc2nc(C)[nH]n2)=O)CC12CCN(C(=O)CC1(CO)CC1)CC2 C1(CC)CNC(=O)CN1C(=O)CN1CC(C)(OC)C1.c12c[nH]nc1CNC2=O C=CC(C)(CCOC)C(=O)NC1CCC(NC(c2cc(F)cc(C)c2C)=O)CC1 c1(C(=O)NC)sc2ncc(CNC3CC3NC(=O)CN3CC=CC3)cc2c1C N1(c2cc(CC)ncn2)CCC2(CCCC2C(=O)Nc2ccc(C)nc2COC)C1 c1(C(=O)NC2CC(F)(CNC(CC(C)OC)=O)C2)c(C)csc1Cl C(=O)(CC1CNc2ccccc21)NC1CN(C(CC(C=C)CC)=O)CC1C c1(-c2c(C)cc(OCC)c(C)c2)ccc2[nH]cc(C(=O)NCc3ccno3)c2c1 Cc1cc(C(N2CC(CCCCNC(c3cnccc3Cl)=O)C2)=O)c(F)cc1Cl C1(NC(c2cccc(C(C)C)c2)=O)CCC2(CCN(C(=O)CC3(C)CC3)C2)C1 C1(F)(C(=O)OC(C)(C)C)CCN(C(c2c[nH]nc2-n2cnnn2)=O)C1 C(=O)(C(C)(C)C(N)=O)NCCCN(C(=O)CC1CCCN1C)CC C1(NC(C2(CC(N)=O)CCC2)=O)CN(C(c2cn(CC(N)=O)nn2)=O)CCC1F CC1C2C(CCN2C(=O)Cc2cnc[nH]2)CN1C(=O)C(O)CC1CCCC1 c1(C(=O)OC2CCC2CSc2ccccc2)cc(Cl)c(Cl)c(I)c1 C1(C(=O)NCCC2CCN(C(=O)CCn3cccnc3=O)C2)CCC(F)(F)C1 C(=O)(CS(=O)(=O)CCO)NCC1N(C(C2C(C)C2C)=O)CC(O)C1 N1(CCCC#C)CCCC(CNC(=O)CCC2CC2(F)F)C1 c1(-c2c(C(=O)NCCN(C(COCCCC#C)=O)C)c[nH]n2)ccc(Cl)c(Cl)c1 C(=O)(C1Cc2ccccc21)NCC1(O)CN(C(c2c(C)cc(Cl)nc2N)=O)C1 N1(C(C(C)OCCCC)=O)CCCC12CCN(C(=O)CN1CCS(=O)(=O)CC1)C2 C(=O)(C1CCC(=O)c2ccccc21)NCC(C1CC1)NC(C(CC)=CCCC)=O C1(CC=C)(NC(=O)C(C2CCCCC2)O)CCN(C(=O)Cn2nc(C)cc2N)C1 c1(CNC(C2(COCC=C)CCCNC2)=O)cc(Br)ccc1I Cn1c(C(=O)NC2CN(C(c3ccccc3)=O)C3CC23)cc(Cl)c1Cl C1(n2cc(-c3c(CNC(CNc4cc(C)[nH]c4)=O)ocn3)nn2)CCCCCC1 C1(NC(C(CC)OCC)=O)CCN(C(C2CC(=O)NC2(C)C)=O)CC1CC C1(C(N(CC)CC2(C)CCN(C(=O)C3CC3)C2)=O)CCCN(S(=O)(=O)CC)C1 C1(N(C(c2cc(C)sc2N)=O)C)CN(C(=O)C(c2ccc(F)cc2)F)CC1(C)C c1(C(N2CC(CC(CN)(C)C)C2)=O)ccc2n[nH]cc2n1.Cn1cnn(CC)c1=O C1(NC(=O)CCN2CCCCC2=O)CC(F)CN(C(c2ccccc2F)=O)C1 c1(C(N2CCCC(NC(C3C(C)(Br)C3)=O)CC2)=O)cc(O)nc2c1CCCC2 CCCCC(CC)C(=O)N1CC(C(=O)NOCC2CCCO2)(CF)C1 N1(C(C(C)Cn2ccnc2)=O)CCC2(C1)CN(C(=O)C(C)(C)F)CCO2 c1(CN(C(C2(C(=O)OC)CC2C)=O)C)cccc(CNC(c2nnsc2C)=O)c1 CCC(CC)C(C)C(=O)NC1COCCC1NC(c1cc(CO)c(C)o1)=O C1(C(N(C)Cc2cn[nH]c2)=O)CCC(O)CN1C(=O)C=C1CCCCC1 C1(N(C(N2CC(C(C)O)C2)=O)Cc2ccccc2F)CCC(C)(C(C)(C)C)C1 C=CCCC(=O)NCC1CCCC1C(=O)NCc1ccc(CO)o1 c1(C(N2CCN(C(C(CC)n3cncn3)=O)CC2)=O)cc2c(cc1N)OCCO2 CC(CC1CCCCC1)C(=O)NCC1CCN(C(c2cnn[nH]2)=O)C1 c1(C(N(CC=CC(=O)NC(COC)(C)C2CC2)C)=O)csc(C)c1 C1(C2CC2)(CNC(c2cnc(C(F)F)s2)=O)CCN(C(=O)Cn2cc(Cl)cn2)C1 N#Cc1cnc2ccccc2c1N1CCC(NC(=O)Cc2csnn2)C1 CC(CC(=O)N1CCC(NC(C2CC(=O)N2)=O)C1C)CC(C)(C)C C1(CCC)CN(C(=O)C(C)P(C)(C)=O)CCN1C(=O)CCOCc1ccccc1 c1(CCC)ccccc1NC(C1CCN(C(=O)C(C2CC2)SC)C1)=O C(=O)(C1=NOC(C)C1C)NCCC1CN(C(c2c(C)nc(O)s2)=O)CC1C c1(OCC)cc(C(=O)NCC2(O)CC(NC(=O)CC3CCCCC3)C2)cc(F)c1 C(=O)(C1=C(C)OCC1)N1CC(SC)C(NC(C2CC3CCC3C2)=O)C1 C1(NC(=O)Nc2ccnn2CC2CC2(F)F)CCn2nccc2C1 c1(C(=O)NCC23CC(NC(CSC)=O)(C2)C3)ccc(-c2cnc[nH]2)cc1 N1(C(c2nc(C)n(C)n2)=O)CCCC2CN(C(=O)C(F)=CC3CC3)CC12 N1(C(C2(C#N)CCCC2)=O)CCC(NC(C2(CF)CCOCC2)=O)C(CO)CC1 C1(CCCC)CN(C(=O)CC2CN(S(=O)(=O)C(F)F)C2)CCN1C(=O)CC#N c1(NC(=O)Cn2nccc2C(=O)NC2CCN(CCF)C2)ccc(F)c(C2CC2)c1 C1(C(=O)NCC2CCC(C(=O)OC)C2)CC2CCC1CC2OC C(CCC1CC1)(C(=O)NC1CCOCC1O)NC(=O)CC1CCC1 N1(CC)CCOC(C(N2CC(NC(c3cncnc3C(C)C)=O)CC2C)=O)C1 c1(C(N2CC3C(CNC(C4CC(=O)NC4)=O)C3C2)=O)coc2c(Cl)cccc12 C(=O)(C(O)C(C)(C)C)N1CCCC(CN(C(=O)CCCC2CC2)C)C1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CC(C(=O)NCc2cnco2)C(O)C1 O=[N+]([O-])c1cc2c(nc1O)CCN(Cc1ccncc1Cl)C2 C1(=CC(=O)NCCSCC(=O)NC(C2CCOC2)CC)CCCC1 N1(C(c2cn(CCOC)nc2C)=O)CCC(CCNC(=O)CC2CSC2)CC1C C1(C(=O)NCC2C(OCC)CN(C(=O)C(F)(F)CO)C2)CCCNS1(=O)=O Cc1sc(C(=O)NCC2CCCC(CNC(=O)C=Cc3cscn3)C2)nc1O c1(CC)cc(C(N2CCCC(N(C(C3CC3(C)C(F)F)=O)CC)C2)=O)cc(O)n1 C=Cn1nncc1C(=O)NCCCN(C(=O)Cn1nccn1)C(C)C O=C(Nn1ccccc1=O)C1CCOCCN1C(c1cc[nH]c1)=O CCC(CC)CC(F)C(=O)NCC1CN(C(c2cnn(CCO)c2)=O)CC1C C1(C(N2CC(C(C)NC(C(C(C)C)CO)=O)C2)=O)CC(c2cccnc2)=NO1 CC1CCC(C)(C(=O)NCCCNC(=O)C=CCN2CCOCC2)C1 C1(CC)(NC(=O)C(CC(C)C)OC)CCCN(C(=O)C=Cc2nccs2)C1 Cc1sc(NC(C)C(=O)O)nc1-c1cn(CCO)nn1.c12ccc(cc1)[nH]c2=O.C(F)F C(=O)(CCC(N)C(C)(C)C)N(C(C)C(c1ccccc1)O)C N1(C(Cc2cccc(C)c2)=O)CCCN(C(c2c[nH]c3ccncc23)=O)CC1C CC1C(NC(c2ccnnc2)=O)CC2CCC1N2C(C1CC2CC(C1)C(=O)N2)=O C1(OC)CN(C(c2nn(C)cc2Cl)=O)CC1NC(=O)CC(C)C1CCCC1 N1(C(c2cc(CSC)c(C)s2)=O)CC2(C1)CN(C(C1(O)CCSC1)=O)C2 c1(CC)cc(C(=O)NC2CCC(NC(=O)COc3ccon3)C2)cc(N)c1 C1(NC(C)=O)CCCN(Cc2ccc(C3(C(F)(F)F)N=N3)cc2)C1 CCC(F)(F)CC(=O)NC1CCC1C(=O)NC1(C(=O)NCC)CC1 O=C(NN1CCCC1C1CCCCC1)C1CCOc2ccccc21 C1(CCCC)CN(C(=O)C(C2CCCC2)OC)CCN1C(c1cscc1F)=O C(=O)(C(C)OCCN(C(=O)C(O)C1CCCC1)CC1CC1)OC.C1(C)CCO1 C1(OC)CN(C(C2(NC(=O)CC(c3ccccc3F)C)CC2)=O)CC1NC(N)=O c1(C(=O)NCC(C(C)C)NC(c2coc(S(C)(=O)=O)c2)=O)cc2c[nH]cnc-2n1 Cc1nc(CNC(=O)CC2(NC(C3CC(O)C(F)C3)=O)CCC2)cc(O)n1 C1(CNC(CC(CC)OC)=O)CCCC2CN(C(=O)CCc3csc(=N)[nH]3)CC12 C(=O)(C1=CCC(C)(C)CC1)N1CC(C=C)C(C(=O)NC2CCc3ncnn3C2)C1 Cc1cc(C(=O)NC2CCC2NC(=O)Cn2cccn2)c(C)n1CC1CC1 c1(C(N2CCN(C(c3cc(F)cc(F)c3)=O)C(CO)C2)=O)cnn2c1NCCC2 C#Cc1ccc(OC)cc1.C1(CCC)C(=O)NC(C)C2(O)CN(C2)CC(=O)N1C C1(NC(C=CC=CCC)=O)CC2CN(C(c3ccnn3CC(F)(F)F)=O)CC2C1 c1(C(N(C(C)C(=O)NCC(Cl)(Cl)Cl)CCC)=O)cccnc1Cl C1(NC(C(C)OCC)=O)CN(C(=O)C=CCn2cncn2)CC1OC C(=O)(C(Cc1ccccc1)C(F)(F)F)N1CCC(NC(C=CCOC)=O)C(O)C1 c1(OCC)ccnc(NC(c2ccc(SC3CC3)cc2)c2nnnn2C2CC2)n1 C(N=c1[nH]cnc(NCC2(COC)CCCO2)c1C)c1nc(NC)sc1 CC1Cc2cc(C(=O)NC(C)CC(C)NC(c3ccc(Cl)cc3N)=O)ccc2O1 C1(NC(C#C)=O)CCCCN(C(C2CC(=O)N(C(C)CC)C2)=O)C1 C(=O)(CN=c1cc[nH]cc1)NCCC1CCCN(C(CCC=C)=O)C1 CC1CC(NC(=O)CNC(=O)Cn2cnc([N+](=O)[O-])c2)CN(C(C2(F)CC2)=O)C1 c1(CC)c(C(=O)N(C2CN(C(C3CCC(O)CC3)=O)C2)C)cnn1CC N1(C(C(CC(C)C)OC)=O)CC2CCN(C(=O)COC(F)(F)C(F)(F)F)C2C1 S(=O)(=O)(c1cccc2cccnc12)N1C(C)(C(=O)NCc2cncc(Br)c2)CC1 C1(CC(F)F)(CN(CCNC(=O)CCCC2CCC2)C2CC2)CCCCC1 C1(C(N2CCC(N(C(C3C(OC)CC3)=O)C)C2)=O)CCc2nc(C)[nH]c2C1 N1(C(C2C(C)CCC2)=O)CCCCC1c1cn(CNC2CC3CC3C2)nn1 Cc1ccc(C)n1CCC(=O)NC(CCNC(=O)CC(C)(C)C)CN(C)C c1(CNC(CCN(C(CCC2CC(C)C2)=O)C)=O)cc(C2CC2)n[nH]1 C1(NC(C2C(C)C2C)=O)CCC12CCN(C(=O)CCC1(C)CC1)CC2 C(=O)(C(C)CCCC(C)=O)NC(CCC#C)C(N1CC(F)(F)C(F)(F)C1)=O c1(OC)ccc(CNC2CN(C(c3cc(I)ccc3Cl)=O)C2)c2ccccc12 CS(=O)(=O)CC1(N(C(C2(c3cc[nH]n3)CC2)=O)C2CC2)CCC1 N1(C(CCCCC)=O)CCCC(C2(NC(C3=CC(C4CC4)(CC)O3)=O)CC2)C1 N1(C(C(N2CCN(C)CC2)C)=O)CCC(NC(c2cc(Cl)no2)=O)C(O)C1 C1(C2(NC(C=COCC)=O)CC2)CCCCN1C(=O)Cc1ccc(O)nc1 C1(CC(=O)NC(c2cccnc2)C)CN(C(=O)CC2(C)CCCCC2)CCO1 Cc1nc(F)ccc1C(N1CCC(F)(C(N2CC(=O)N(C)C2)=O)C1)=O c1(CC(=O)NCC2(COC)CCN(C(=O)CC(C)F)C2)c(C)cccc1F N1(C(C2C(C)C2)=O)CCC(c2nnc(CNC(=O)COC(F)F)s2)CC1 CCCCC(O)C(=O)N(C1CC12CCNCC2)c1cc(C2CC2)ncn1 CN1CCN(C(=O)C(C2CC2)NC(c2cccc(O)n2)=O)C(CO)C1 N1(C(COC(C)=O)=O)CCCC2CN(C(c3nccnc3N)=O)CCC12 c1(OCC(C)C)ccc(NC2(c3nnnn3C(C)C)CSCC2C)cc1 c1(C(=O)NC2CC(NC(C3CC(=C(F)F)C3)=O)C2)ccc([N+](=O)[O-])o1 C(C)(CC(C)N=c1[nH]c(Cl)ncc1OC)NC(CC(CC)O)=O c1(OC)ccc(F)c(CC(=O)NCC(C)(C)CNC(c2[nH]c(=N)ccc2C)=O)c1 C=CC(C)C(C)C(=O)Nc1cccc(NC(c2cc(Cn3cccn3)on2)=O)c1 c1(C2(C(N(CCOC)CC)=O)CC2)ccc2c(c1)OCO2.c12csc(C)c1O2 CC(C)(C(F)(F)F)NC(C1CCCC1n1cc(C2CC3(CCC3)C2)nn1)=O C1(C(=O)NC(C(=O)NCCCS(C)(=O)=O)CCOC)CC12CCOCC2 C1(c2ccc(F)cc2)(NC(C2C(COC)C2)=O)CCN(C(c2conc2C)=O)CC1 c1(C(N2CC(NC(C(CC)SC)=O)C(OC)C2)=O)c[nH]c(=N)c2[nH]ccc12 N1(C(C2CCCN(CC(C)C)C2)=O)CCC(NC(c2ncc[nH]c2=O)=O)C12CC2 C1(CNC(COCCC#C)=O)C2CC1N(C(=O)CSCC(C)C)C2 Cc1cccc(C(N2CCCCC2CC(=O)NCc2ncco2)=O)c1N C(=O)(CCCCC(N)=O)N1CC(CNC(Cc2cc(OC)c(O)cc2)=O)OCC1 C1(C2(O)CN(C(c3c(C)noc3C3CC3)=O)C2)(CNC(C)=O)CC1 C(=O)(C1=CCCC1C)N1CCCC(CCNC(CC(CC)c2ccccc2)=O)C1 S(=O)(=O)(c1cc(Br)ccc1F)N1C(C)CSCC1.c12cccc(c1)N2 C1(N(C(c2cnc(C)[nH]2)=O)C)CN(C(c2ccc(F)c(Br)c2)=O)CC12CC2 Cc1ccc(CSC(C)C(N2CCCC2CN(C(=O)C2=COCC2)C)=O)cc1 N1(C(C2CC(CC)(CC)C2)=O)CC(CNC(=O)COC2(C)CCC2)CC1C C1(C(=O)NC(C2CCC2)C)CC2(CC(NC(C3CC4(CCO3)CC4)=O)C2)C1 C1(N(C(C(C2CCC2)OC)=O)C)CN(C(C23CCCC2C3(F)F)=O)CCC1O C(=O)(C(C)CSC)NCC1CC(NC(C2CC(C(=O)OC)C2)=O)C1.C(C)(C)(C)N c1(NC(C2CC3CC3N2C(c2cnc(Cl)c(I)c2)=O)=O)cc(Br)ccc1O C1(C(N(CC(CC)(C)OC)C)=O)CC(F)(F)CN1C(c1cc(O)nc(O)n1)=O c1(OC)cccc(NC(c2ccc(C(C)NC(=O)C(=O)NCCSCC)s2)=O)c1 C(=O)(C(C)CC(C)(F)F)NC(CCCC)CNC(c1cc[nH]n1)=O C1(NC2(c3nnnn3CC3CCCO3)CC(C=C)C2)Cc2ccccc2C1.C1CC1 c1(C(N2CCC(F)(F)C2)=O)cccc(COC)c1F.N12CCCC(C1)C2 C(CCCO)N(C(=O)CNC(=O)CNC(=O)COC1CCC1)CC CC(C)C(CNC(=O)C(O)CCNC(=O)CN1CCC(C)CC1)CO C(C(C(=O)NCc1cccnc1)NC(=O)CC1CCCO1)OC(C)C c1(C(N2CC(N(C(C(C)Cc3cnc[nH]3)=O)C)C2)=O)ccc2nc(O)oc2c1 C1(C(N2CC(O)(CCNC(COCCC)=O)C2)=O)CC12C(=O)Nc1ccccc12 Cn1cccc(C(=O)NC2CCCC2NC(c2cc(Br)ccc2O)=O)c1=O CCC(CC)(CN=c1cc[nH]cc1[N+](=O)[O-])NC(C1CCC(=O)NC1)=O C1(CNC(c2ccc(C)cn2)=O)CC2(CCN(C(C3CC4(CC4)C3)=O)CC2)CO1 N1(C(C(C2CCOC2)OC)=O)C2CCC1CN(CCC1CCCC(C)C1)CC2 C1(C(=O)O)CC(O)C12CCC2.C(CCCNC(=O)CSCC(F)F)N(C)C c1(C(=O)NCCCn2cc(C3CCN(C)C3)nn2)c(F)cccc1[N+](=O)[O-] Cc1c(CC(=O)NCC2C(C(N3CCCC3CF)=O)C2(C)C)ncn1C C1(N(C(c2c(C)nc[nH]2)=O)C)CCCC(N(C(=O)Cc2ncsc2Cl)C)C1 C1(N(C)C)CCCN(C(=O)CCn2cc(COc3ccccc3Cl)nn2)C1 C123CCCN(CC1C2)C(=O)C(N(CC)CC)CCSCC=CC(=O)N3.CC.SCCC c1(CC(=O)N(C(C)CCNC(C2CC23CC3)=O)C)c(Br)ccc(F)c1F C(=O)(C(C(C)(C)C)SC)NC(CC)CNC(c1ccc(C)o1)=O c1(CNC(C2CC(C)C2)=O)ccc(C(=O)NCc2ccc(C3CC3)cn2)cn1 N1(C(c2cn(C(C)C)nc2)=O)CCC(C)C(NC(=O)Cc2n[nH]c(=N)s2)C1 Cc1cc(C(=O)NC2CCC(CCNC(=O)C(=O)Nc3ccccc3)C2)ccn1 C#CCC(C)(C(=O)N1CCCC(CC)C1)NC(=O)C=Cc1cncs1 C12CC13CCN(C3)C2=O.c1(CNS(CC)(=O)=O)cnc(O)c(C)c1 C(=O)(C(O)CC(C)C)NCC(CC=C)NC(c1ccc(=O)n(CC)n1)=O C(=O)(C(O)CC(F)(F)F)NCC(N(C(=O)CCCC1CCOCC1)C)C1CC1 C1(C(=O)NCc2cc(OC)c(OCC(=O)N(C)C)cc2)CN2CCCC2CO1 C(=O)(CCCC(=O)NC1CC(C)N(C(C2CCCC2C)=O)C1)NC N1(C(C(CC)OC)=O)CCc2c(c(CNC(C3(CNC(C)=O)CC3)=O)nn2C)C1 C1(CN(C(=O)CC2CC(F)C2)C)CC2(CC2)CN1C(=O)C=CC(C)(C)C CC1CCC(C)N1CC(=O)NCCC(C)(C)N(C)C.C1C(F)C(=O)N1 CCC(C(C)CN(C)C)NC(C1(NC(=O)CCn2cncn2)CSC1)=O c1(CCCC(=O)NCC(CC)(C)NC(c2cc(Cl)c[nH]2)=O)ccc(OC)cc1 N1(C(C2N(C(=O)OC)CSC2)=O)CC2CC1CN(C(C1CCS1(=O)=O)=O)C2 C12(C(=O)NC(c3c(C)n[nH]c3C)C)CCC(NC(C3CC3C3CCC3)=O)(CC1)C2 c1(C(N2C(c3cn(CCOC)nn3)CC2)=O)cc(C)nn1CC(F)(F)F c1(CNC2CCCC(C(=O)Nc3cn[nH]c3)C2)c[nH]c2ncc(Cl)cc12 c1(OC)cccc(C2CCCN(C(=O)Cc3cn(C)nc3C#N)C2)c1F CC1(C)CCCOC1CC(N1CCCCC(CNC(c2n[nH]c(O)n2)=O)C1)=O n1(CCC)cc(-c2cn(C(C)CN(C(c3cc(C(C)C)[nH]n3)=O)CC)nn2)cn1 N1(C(Cc2c(C)occ2)=O)CCOC2(CCN(C(=O)CCCc3cnn[nH]3)C2)C1 Cc1cccc(C(=O)NC2(CO)CCN(C(C3CN4CCN3CC4)=O)CC2)c1O c1(C(=O)NC2(COC)CCN(C(C(CC)F)=O)CC2)nc2ccccc2cc1Cl C1(NC(C(C)OC2CCCC2)=O)C2CC3C(C2)C13C(=O)NCCC(O)C1CCC1 N1(C(C(CCN(C)C)O)=O)CC2CCC1C(C(=O)NC1CC3C(C1)C3(C)C)C2 CCCCCC(O)CC(=O)N1CCCN(C(c2ccc(O)c(C(C)=O)c2)=O)CC1 c1(C(N(C2C(C)CCN(C(C)=O)C2)C)=O)cc2c(Br)coc2cn1 c1(C(N(C2CCCN(C(CC(CCC)C)=O)C2)C)=O)cc(OC)c(OC)cc1C Cc1sc(C(N2CCC(F)(CNC(c3occc3Br)=O)C2)=O)c(C)c1C c1(CC(N2CCC(CNC(=O)C(F)(F)CO)C2)=O)c(F)cccc1F C12(CC(N3CCC(N(C(=O)C(O)Cc4ccccc4)CC)C3)=O)COC(CF)(C1)C2 C12CC(=NO1)C(=O)NC2.C1(=O)CC1=O.C1(CN)CC2CC2C1.CNC Cc1cc(C)c(C(=O)NCC2CN(C(=O)C=CCN(C)C)CCC2C)cc1C Cc1cncc(C)c1C(=O)NC1CC1NC(=O)C(F)(Cl)c1ccccc1 c1(C(=O)NCC2CN(C(c3cc(CCC)[nH]n3)=O)CC2O)cc2c[nH]cnc-2n1 N1(C(CN2CCC(OC)C2)=O)CCC2CN(C(c3c(SC)cccc3F)=O)CC12 CC1CC(C(=O)NC2(CNC(c3cncc(N)c3)=O)CCC2)CC(C)(C)C1 c1(CC(=O)NC(C)C(CO)NC(=O)CC(C)C(C)(C)C)ccc([N+](=O)[O-])cc1 CC(C)(C)CCC(=O)N1CC(CCNC(c2cocc2C(N)=O)=O)C1 N1(C(c2c(Cl)cn(C)n2)=O)CCCC(NC(=O)CCCOc2cccnc2)CC1 CCC(CN(C)C)CC(=O)NCc1cccc(C(=O)NCCN2CCC(C)C2)n1 c1(C(=O)Nc2cncc(C(N3CCC(OC)CC3)=O)c2)cc(C)cc(Br)c1F c1(C(N(CC(=O)NCCC(C)O)CC#C)=O)oc(C)nc1C c1(CC(N2CC3C(CNC(CCCCCOC)=O)C3C2)=O)ccc(S(C)=O)cc1 O=C(C1CCCc2nn[nH]c21)NC1CCSC12CN(C(C1(CO)CCCC1)=O)C2 C#CCC(C)(C(=O)N1CCCC(NC(N)=O)C1)NC(c1n[nH]c(C)c1C)=O c1(C(=O)NCC2CCN2C(=O)CC2CC2C(F)(F)F)ccc(Cl)c(Cl)c1 c1(C(=O)NC2(C)CCN(C(C(c3ccc(C)s3)C)=O)C2)n[nH]c2c1CC(C)(C)C2 c1(C(=O)NC(C(C)NC(C2CC(F)CN2C)=O)CO)cn2ccc(F)cc2n1 c1(OCC)ccc(C)cc1.C1(N(C(C)CNC(=O)COC)C=O)CC12CC2 c1(OC)ccc(C(=O)NC2(C3CCCN3C(C3C4CCCCC34)=O)CC2)cc1 C1(C(=O)NCCC2CCCN2C(c2cc[nH]c2C2CC2)=O)CCC(C(F)F)CC1 N1(C(Cn2ncc(C)c2)=O)CC2CCN(C(=O)CC3CCCNC3=O)CC12 N1(C(C(CCC)NC(C(CCC)NC(N)=O)=O)=O)CCC(C2CC2)CC1 c1(NC(C2CC3CC3N2Cc2ccnc(OC(F)F)c2)=O)cc(F)c(F)cc1Br CN1CCC(Cc2cccc(Cl)c2)(CNC(=O)CN2CCS(=O)CC2)CC1 Cc1cc(N2CCC(c3n[nH]c(C)n3)CC2)c(O)nn1 c1(OC)ccc(C(=O)N(C2CN(C(=O)Cc3cccc(C(F)F)c3)C2)C)cc1O C(=O)(C(C)CC(=O)c1ccccc1-c1ccc(C)cc1)OCC(C(=O)OC)C C(=O)(C(C)(CO)NC(c1cccnc1S)=O)NCC(C)OCCO C1(C(N2CCN(C(c3n(C(C)C)ncc3)=O)C(CF)C2)=O)CCC2(CCC2)OC1 C1(COC)CN(C(c2cc[n+]([O-])cc2)=O)CCN1C(c1cncc(N)n1)=O C(=O)(C(F)C(F)(F)F)N1C(C)CC(CNC(c2cccc(Cl)n2)=O)C1 N1(C(C(C)(CO)NC(c2cncc(C#N)c2)=O)=O)CC2CCC1C(O)C2O N1(C(=O)CC2CC3CCC2O3)CCC2(CC1)CN(C(=O)CC1CCCO1)CCO2 C1(C(=O)NOCC2CCCC2)CCOCC1NC(C1(CC2CC2)CC1)=O N1(C(CCc2onc(CC)n2)=O)CC2COCC2(C(=O)NC(CC)C(F)(F)F)C1 N1(C(C(C)C)=O)CCN(C(=O)COc2cccc(C3CC3)c2)CCC1C c1(NC(C2CC23CCN(C(=O)CC2CCC2)C3)=O)cnc2ccoc2c1 N1(C(C)=O)CCC(F)(C(=O)NCCOCCOCCN(C)C)C1.c1cc(CO)no1 c1(C(=O)NCC2CCN(C(c3ccc(COC)[nH]3)=O)C2)c(Cl)ccc(O)c1N N1(CCNC(NC(c2nccs2)C)=N)CCCCC1 c1(C(N2CCOCC2)C(=O)N(CC(C)C)CC2CCCOC2)scnc1C(=O)OC c1(CC)c(C(=O)N(CC(C)(C)NC(C2CC3CCC2C3)=O)C)csc1C S1(=O)(=O)c2ccc(cc2C(C)C)N1CC.C(=O)(CCC(C)SC)O.CCO c1(C(=O)NCC(C)N(C(=O)C(F)C(F)(F)F)C)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 N1(C(c2c(C)oc(CC3CC3)c2)=O)CC2CC1CN(C(c1cn(C(C)C)nn1)=O)C2 N1(CCC(=O)NCCCCC(C)NC(CCCC(=C)C)=O)Cc2ccccc2C1 c1(CC(=O)NCC)ccc(N2CCN(CC3C(NC(CCC=C)=O)C3)CC2)cc1 c1(C(=O)Nc2ccc(C)cc2Br)cc(-c2cnn(C(C)C)c2)c2cn[nH]c2c1 C(C)(C)(CC(F)C(=O)NC1CSC1)NC(CC(COC)(C)C)=O CC(C)CC(O)C(C)C(=O)N1CC(C(C)NC(=O)CCSCC(C)C)C1 c1(OC(C)C)ccc(C(=O)NC2CC2C(=O)NCc2ccc(Br)nc2)c(F)c1 C1(NC)CCCC(C(=O)Nc2ccccc2OC(COC)OC)C1 c1(C(=O)NC(C(=O)NC2C(C)CCC2)Cc2ccoc2)cnn2c1OCC2 Cc1nn(CC(=O)NC(C)CCNC(C2CCCN2c2nccs2)=O)c(C)c1C C1(C)(C(=O)NCC(CNC(COCCSC)=O)C)Cc2ccccc2C(=O)O1 C(=O)(C(Cc1ccccc1)CC(C)C)NCC(C)N(C(COCC)=O)C N#Cc1cc(NC(C2CSCCN2Cc2cc(F)cc(Br)c2F)=O)cc(F)c1F N1(c2scc(C)n2)CCC(C(=O)Nc2ccccc2OC(C)(C)C)C(C)C1 CC(C)C(C)C(=O)N(C1CCCCC1N(C(=O)CSc1cnn(C)c1)C)C Cc1ncc2n1CCN(C(=O)CC1(NC(c3cn(C)nn3)=O)CC1)C2 Nc1ccc(C(=O)NCC2CCCC(NC(=O)Cc3ccccc3)C2)c(O)c1Cl C1(C(N(CC(=C)C)C)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC1(C)C N1(C(c2c(CC)onc2)=O)CC(N(C(=O)Cc2ccc(Cl)c(F)c2)C)C2(CC2)C1 CC(O)CCCN=c1[nH]c(=NCC2CC23CCC3)c2c(F)cccc2[nH]1 c1(C(=O)NCC(C)CNC(C2(C3CCCO3)CCC2)=O)c(O)cc(Cl)cc1Cl CC1=NOC(=O)C1CCC(=O)NCC1(F)CN(C(c2ccc(C(C)(C)C)o2)=O)C1 C1(NC(C2C(=C)C2)=O)CC2(CCCCN2C(=O)C(CC)N(CC)CC)C1 C1(C(=O)NCC2(CNC(c3c(CC)n(C)nc3)=O)CC2)CCOCC12CCC2 c1(CNC(c2cn[nH]c2)CC)cc2cccc(F)c2o1 N1(C(CN2CC(C)C2)=O)CCN(C(=O)C(c2cccnc2)C)CC1C(C)(C)C C1(CC)CCCN(C(C2CCC2C(C)(C)C)=O)C1C(=O)NCC1COCC1(C)C c1(C(N2C(CNC(c3c(C)nsc3N)=O)CC2)=O)cccc2c1ncn2C C1(C(=O)NC(C(=O)N(C)CC2CC2(C)C)(C)C2CCC2)CC(C)(C)CCO1 c1(CNC(N2CCOCC2c2nc[nH]n2)=O)ccnc(F)c1F CC(C)CC(C)C(C(=O)NCc1ccc(F)cc1)N1CCC(CCCO)CC1 N1(C(c2oc(C)c(Br)c2)=O)CCN(C(c2ccc[nH]2)=O)C(CC(F)F)C1 C(C(C)N=c1ccnc(CC)[nH]1)(c1ccccc1)NC(CC(CCC)O)=O N1(C(C(CC)C(C)C)=O)C2CCC1CC(CNC(=O)C=CC(C)(C)C)C2 Cc1cncn1CC(=O)NCCSCC1(C2CCOC2)CC1 N1(C(C(C)(O)C2CCOCC2)=O)CCC(C)(NC(=O)C(c2ccccc2)F)C1 c1(OC)ccnc(C(N2CCOC(C(=O)Nc3cncc(Cl)c3C)C2)=O)c1OC C1(NC(CCC(=O)NCCC)=O)CC2(CCN(C(c3cccnc3F)=O)CC2)C1 c1(CN2C3C(C3C)C2=O)cc(N)cc(F)c1.c1(C(=O)OC)ccc(C2CC2C)o1 n1(CCOC)cc(CN2CCC(NC(=O)C(C)OCC)C2)nn1 C1(=O)C(O)C(C(C)C)NC2CCCN1CC2.N1(CCCCOC)CCNCC1 C1(NC(CC)=O)CC12CCC(NC(c1cccc([N+](=O)[O-])c1)=O)CC2 c1(C(=O)NCC(C)N(C(=O)Cc2ccnc(F)c2)C)cc(=O)c2ccccc2o1 c1(NCC2ON=C(C)C2)cc(OC2CCOCC2)ncn1 CC1CCCCC1CC(=O)NCCOC1(CNC(=O)CS(N)(=O)=O)CCOCC1 Cc1cc(F)ccc1C(N1CCN(C(C2CCCN2C=O)=O)CC1CC(F)F)=O C(=O)(CCCCCF)N(C)Cc1ccc(CNC(CN(C)C)=O)cc1 n1(CC)cc([N+](=O)[O-])c(C(=O)N(C)CCN(C)C(C2CC2C(C)C)=O)n1 c1(CC)cccc(C(=O)NCCC(O)CNC(c2cc(C(N)=O)c[nH]2)=O)n1 c1(CN2C3C(C(=O)N=c4[nH][nH]cc4Br)C(C3)C2=Cc2ccccc2)cnc2cc(Cl)ccn12 C(C(=O)NCC1CN(C(=O)CSCC(C)=O)CCO1)(C(C)C)SCC c1(C(=O)NCC(C)NC(c2c(C(=O)OC)cccc2)=O)ccnc2ccncc12 C1(C(=O)NCC(C)(CNC(=O)C(O)C(F)F)OC)CC(O)CN1C(N)=O N1(C(C2(OC)CCCOC2)=O)CC2(CCN(C(c3ccc(F)c(F)c3C)=O)C2)C1 C1(COC)(CNC(=O)C=C(C)c2ccsc2)CCN(c2cc(C)nc(C)n2)CC1 C(=O)(CC(=O)NC(C1CCCC1)CNC(C1CSC1)=O)OCCC(C)C Cc1cnc2nc(C(=O)NCCOCCNC(=O)C(C)(C)C)nn2c1 c1(C(=O)NC2CCC(N(C(c3cc(OC)no3)=O)C)C2)cccc2occc12 N1(C(CN(CCC#C)C)=O)CCC(CNC23CC(CC(C)C)C2C3)C(C)C1 O=C(CS(=O)CCC(F)(F)F)N1CC2CCN(C(=O)C(F)=CCCF)C2C1 CC(C)(C)C(C(=O)NCCCCCNC(C1CCCO1)=O)N1CCNC1=O N1(C(C2N(C(CC(C=C)C)=O)CC(O)C2)=O)CCOC2COCC2C1 c1(C(=O)NC(CC=C)CNC(=O)CCC2(C)CC2)cc(C(C)C)oc1C(C)C C(C(=O)N(CC(=O)N(CCCC)CC1CC1)C1CC1)=CC=C.C1CN1 C1(C(C)(C)C)CCC(C(F)(F)F)N(SC2CCC2)C1 c12ccc([nH]1)C2.C(CC(=O)NCC1CC1NC(=O)Cc1cccs1)N(CCC)C c1(CC(N2C(C(=O)OCC)(CC)CC(N)C2)=O)c(C)nc(C(C)CC)nc1C C1(C(N(CC(=O)NCCC)C)=O)CCCN1C(=O)C(C1CCC1)OCC N1(C(C(C)CN(C)C(c2coc(N(C)C)n2)=O)=O)CCC(C)(C)C(CO)C1 c1(C(N2C3CC(CN(C(CCCCC)=O)C3)C2)=O)ccc2c(c1)NCC(=O)N2 C1(NC(=O)CCc2ccc(Cl)s2)CC(NC(C2CC3CCC2O3)=O)CC1O CCCCC(C(=O)NC(C)CCNC(c1ccc(CC)[nH]1)=O)N(C)C CCCC(CC(=O)NCCc1ccns1)NC(=O)CN1CCOCC1=O C1(CC(=O)N(CCCNC(COCC#C)=O)C(C)C)C(=O)NN=C1C C(=O)(CCc1cccs1)N(C(CNC(=O)Cc1nncs1)C1CC1)C N1(C(CC(C(C)O)N)=O)CCCC(C2CC2NC(=O)C(F)(F)F)C1 Cn1nc2ccccc2c1C(=O)NCC1(NC(C2(Cl)CC2)=O)CCCCC1 C1(CNC(C(CCC)C)=O)CC2CCC(C1)N2C(C1CC(C2CCC2)=NO1)=O Cc1cc(C)n(CC(=O)NCC2(F)CCC(NC(c3nnn(C(C)C)n3)=O)C2)n1 C1(NC(C2(C)CCNC(=O)C2)=O)CC2(CCN(C(c3cccc(O)c3F)=O)C2)C1 C1(N(C(CN(C(=O)OC)C)=O)C)CCC(NC(=O)CCn2cc(C)cn2)C1 N1(C(C(C)OC)=O)CC(CN(C(=O)CC(=O)N(C)C)C2CC2)C2(CC2)C1 CC#CCC(C(=O)NCCN1CCCCC1)NC(=O)CN(C)C(N)=O C(CCC(=O)NCC1(NC(=O)CC2CCCC2C)CCC1)OCC=C c1(OCCC)ccnc(CCN(C(C)=O)Cc2conc2-c2ccccc2)n1 C1(CC=C)(NC(C2(C)CC2c2ccccc2)=O)CCN(C(=O)C(CC)OCC)C1 c1(C(N(C2CC(NC(=O)CC3SC(=N)NC3=O)C2)C)=O)csc2c(O)ccnc12 c12cccn3c(cnc13)C(=O)OC2.CC1OC2(C)CC1(C(=O)N(C)C)C2 C1(C(=O)NCC(NOC)=O)CCN(C(=O)CCCC2CC2C)C12CCC2 CC1(C)CC(NC(=O)C(C2CCN(C(=O)CC3CCCC34CC4)C2)F)CC(O)C1 c1(OCCOC)cccc(CCC(C)NC(=O)NCCCC2(C)OCCO2)c1 C12(C(=O)Nc3nc(CNC(=O)CCCC4CCCC4)oc3)CCCCC1OCC2 c1(C(=O)NCCC(CCNC(c2c(C)scn2)=O)C)cc2c(O)ncnc2cn1 CON(CCC(=O)NC(C)CCc1ccco1)C(=O)C1CCN(C)C1 C1(C(=O)NCC2(NC(C(CCC)C)=O)CCCC2)CS(=O)(=O)CC12CC2 Cc1cc(C)n2ncc(C(N3CCN(C(=O)CN4CC(C)C4)C4CC34)=O)c2n1 Cc1nn(C)c(C)c1C(=O)C(N1CCC(NC(c2scnc2C(C)C)=O)C(O)C1)=O N(C(=NCCC1(C)OCCO1)NC(C)C)C1CC(OC)C1(C)C C1(C(=O)NC(C(C(=O)OC)C)C)C(C2CC2)CCN1C(C1CCC1)=O c1(C(=O)NC2CCC(NC(=O)C(O)Cc3cnc[nH]3)C2)ccn2c1CSCC2 C1(C(=O)NC2C(OC)CN(C(=O)CCCC(=O)C3CC3)C2)CN2CCN1CC2C CC1=NC(C)(CCNC(C2CCCCC2NC(=O)C2CC2)=O)CS1 C1(NC(=O)NC(C(C)OC)C)CCSC2(CCC2)C1 CC1CC=CCC1C(=O)NCC(c1cccc(Cl)c1)NC(C1(F)CCCC1)=O c1(CNC(C(N(C)CP(C)(C)=O)=O)=O)cc2c(cn1)CCCC2 C1(C(=O)NC(CC=C)CNC(=O)CCn2cccn2)CC2(C1)CC21CC1 N1(C(C2=NOC(C)C2)=O)CCC2CCC(NC(C3CCC(C(N)=O)CC3)=O)C1C2 c1(C(N(C(CNC(=O)C(O)CF)C2CC2)C)=O)cnn(C(C)(C)C)c1 C1(NC(C(F)=CCC)=O)CCC2CN(C(c3cncc(N)c3C)=O)CC2C1 C1(NC(C=C(C)Cl)=O)CCCCC12CCN(C(C1(F)CC3(CCC3)C1)=O)C2 CC1(C(N2CCOC(C(=O)NC(CO)C3CCC3)C2)=O)C=CCCC1 C1(CNC(c2c(C(C)C)n[nH]c2)=O)CC(NC(=O)CCc2cncn2C)C1(C)C C(CC(F)F)(C(=O)N1CCC(C2CCCO2)C1)NC(c1ccsc1)=O N1(C(c2ncsc2C2CCCC2)=O)CCCN(C2COC2)CC1 CNS(=O)(=O)c1ccc(C(N2CCC(NC(C3(C(C)C)CC3)=O)C2)=O)cc1 N1(CC)CCCC(N=c2[nH]c3c(c(=NCc4ccnc(C)c4)[nH]2)CSC3)CC1 C1(NC(c2ccc(COC)o2)=O)CCOC(C(=O)NCCc2nccc(O)n2)C1 C=C(CNC(C1CC=CC(NC(C2CCCCN2C)=O)C1)=O)C(F)(F)F C(C)(C1=CCN(C)CC1)NC(C1N(C(CN(CCC)C)=O)CCOC1)=O C(=O)(CCCC(N)=O)N(CC(CO)(CO)NC(=O)CC1C=CCC1)C Cc1cc(N2CCCC(NC(=O)CCn3ccnc3)C2C)ncc1[N+](=O)[O-] N1(C(C(C)NC(CC)(C)C)=O)CCCC1(C)CNC(=O)CCc1ccc(C)cc1 C1(OC)CN(C(=O)CCC2CCCC2)CC1NC(c1c(C(C)=O)cnn1C)=O c1(C(N2CC(CNC(c3n(CCC)ncc3)=O)C(C)C2)=O)cccc(C#N)c1C C(=O)(C1CCCc2ccccc21)N1CCC(C)N(C(=O)CC2CCOC2)CC1 N1(C(c2ccc(CC)cn2)=O)CCOCC1(CO)CC C(=O)(CCC(F)(F)F)N1C(CCC(=O)N(C2COCC2O)CC)CCCC1 CC1CCN(C(c2cc(C(N)=O)ccn2)=O)CCN1C(=O)CC1CCC2CC12 C#Cc1cncc(C(N2CC(NC(C3(c4cccs4)CC3)=O)CC(C)C2)=O)c1 N1(C(C2C3(N(C(C(C(C)(C)C)O)=O)CC3)C2)=O)CCc2ncccc2C1 C(C(C)CC(=O)N(CC(C)CO)CC)NC(C(C(C)C)OCC)=O CN(Cc1cc(C(F)(F)F)n[nH]1)N1CCCC(Cn2ccnn2)C1 c1(C(=O)NC(C)C(CO)NC(c2[nH]nc3ncccc23)=O)cc2c(s1)COCC2 c1(C(N(CC(C)NC(C=C(CC)C)=O)C)=O)scc(N)c1C C=CCC(CNC(=O)CSC1CC1)C(=O)NCc1ccc(OC)nc1 c1(C(C)C)ncc(C(=O)NC2(C)CN(C(C3CC3c3cccs3)=O)C2)n1C C(=O)(C(C)(C)CC1CC1)NC(CC(C)NC(c1ccc(Cl)cn1)=O)C N1(c2cc(C)nc(NC3CCOC(C4CC4)C3)n2)CCc2c(nnn2C)C1 Cc1cc(C(=O)NCC(C)NC(C2CCC(C(C)C)CC2)=O)[nH]c1C c1(CC(=O)NCCOCCN(C(=O)CSc2ccccc2F)C)cc(Cl)n(C)n1 N1(C(CC(C)C(C)(C)C)=O)CCOC2CCN(C(C3(C(N)=O)CCC3)=O)CC12 C(CCC(=O)Nc1ncn(-c2ccccc2)n1)OC(C)=O C1(c2nc(CC)[nH]n2)CC12CC(C(=O)NCCN1CCCC1C)C2 N1(C(Cc2n(C)cnc2)=O)CC2CC1(C(=O)NCC1CC(C)(O)C1)C2 Cc1nc(NC(C2(C)CCCN2C(c2cccc3[nH]ncc23)=O)=O)c(C#N)n1C N1(C(C2(CC=C)CCC2)=O)CC(NC(=O)CC23CCCC2C3)C(O)C1 c1(C(=O)NC(CC(C)NC(c2c(C)noc2)=O)C)cncc2[nH]ccc12 C=CCC(C)C(=O)N(C1CCCCC1)CCNC(c1cn(CC(F)F)nc1C)=O C=CCC(CC)C(=O)NCC1(F)CN(C(c2ccnn2CC)=O)C1 Cc1nc(C)c(CC(=O)NCC2CCN2C(c2cnc(C3CC3)[nH]2)=O)s1 N(C(=NCCS(=O)(=O)N1CCCC1)NCCNc1cccc(C(F)F)c1)C(C)C N1(C(C(C)CO)=O)CC(O)C(O)C1 C=CCC(CC(=O)NCC1(CO)CC1)NC(=O)CC1CCOC1=O c1(CCC(=O)NC2CC(N(C(C(C)SC3CC3)=O)C)C2)cnc(C2CC2)o1 C(C1CCCCCC1)=CC(=O)NC1(CNC(C23CCCC2CC3)=O)CCCCC1 CCCCCC(=O)NCCN1CCC(NC(=O)CCn2cnccc2=O)CC1 C1(C(=O)NC(C(C)C)CCNC(=O)C(C)(C)C2CCC2)CN2CCC1(C)CC2 C#Cc1cccc(C(N2CCC(C3CC3)(NC(=O)CC3CC3)C2)=O)c1Cl c1(C(=O)NC(CNC(C(CC(C)C)O)=O)CC(F)(F)F)noc2ccc(Cl)cc12 C1(OCC(=O)NCC(C)(C2CCC2)NC(=O)C=CC2CC2)CCOCC1 N1(C(C2C(C)CN(C(C3CC34CCOCC4)=O)CC2)=O)CC(C)N(C)C(C)C1 c1(C(=O)NC2CN(Cc3c(F)cc(OC)c(F)c3)C2)cc([N+](=O)[O-])c(C)cc1F N1(CCS(=O)(=O)NC)CCCC(C(F)(F)F)(Nc2ncc(O)cn2)C1 C(=O)(C1CCCc2ncccc21)NC1CC(C)(NC(CCC#C)=O)C1 C1(C(=O)NCCNC(C2C3C4CCC(C4)C23)=O)CCc2ccc(F)cc2O1 n1(CC(=O)NC2C(NC(C(CC)O)=O)COC2)ncc2ccc(OC)cc2c1=O CC1(NC(=O)CC(F)(F)Br)CCN(C(c2ccccc2OCCF)=O)C1 c1(C(=O)NCC(CCCC)NC(=O)CNC(N)=O)c[nH]c2cc(Cl)ccc12 C1(NC(=O)NC(c2cc(F)cc(Br)c2)C)CCOC2(CCCC2)C1 C(C)(C(C(=O)N1CCC(OCCOC)C1)NC(C1C=C(C)CS1)=O)OC c1(C(N2CCCC(C)(OCC)C2)=O)nc(=NC(C)c2ccccc2)cc[nH]1 c1(C(C(=O)NC)N(C(c2ccccc2)C(F)F)C)c(Cl)cnn1C c1(C(=O)Nc2cn(C)nc2)cccc(S(=O)(=O)NCCNC(C2CCCO2)=O)c1 CCCCCCCCCCC(=O)N1CCN(C(C2CCCNS2(=O)=O)=O)C(C)C1 c1(C(N2CCC(CN(C(C3N(CCC)CCC3)=O)C)C2)=O)c(F)ccc(N)c1F C12(CNC(c3cnn(CCF)c3)=O)CCC1CN(C(C1(O)CCOCC1)=O)C2 c1(C(N2CCOC(C3CCOCC3)C2)C(=O)N(C)C2CC2)c2c(nn1C)CCOC2 N1(C(C(C)OCC)=O)CCCCC1C1CCCN1c1nnc(COC)s1 c1(CC(N2CCC(NC(CN(CC)CC)=O)C2C)=O)c(C)nn(C(C)C)c1C Cc1cnncc1C(=O)NCC(CO)NC(C1CCC(O)CC1)=O C(=O)(CC(C)(C)C(=O)N1CCCCC(C(=O)NCC2(N(C)C)CCC2)C1)OCC CC1CN(C)CC1C(=O)NCC1(F)CC(NC(=O)CN2CCCCC2)C1 C(C(=O)NC1CC(C)(CNC(=O)CC2COCC2(C)C)C1)(C(C)C)NC(C)=O Cc1cc(C(=O)NC2CCC(CCNC(=O)CNc3ccccn3)C2)cn1C CC(C)C(CNC(C1(CO)COC1)=O)NC(=O)Cc1cncn1C c1(C(=O)NC2C(NC(C3CN(C(C)=O)C3)=O)CCC2)cc(SC(F)(F)F)oc1C Cc1ccc(C(N2CCN(C(c3[nH]nnc3C3CC3)=O)CC2CC2CC2)=O)nc1C c1(OC)ccc([N+](=O)[O-])cc1CN1CCC(C(N2CCC(C)C(O)C2)=O)C(O)C1 N1(C(C(CC#C)(C)C)=O)CCC2(CC1)CC2C(=O)NC1CCC2CCC12 C1(CNC(C2(OC)CC2)=O)CCCCN(C(c2ncccc2CSC)=O)C1 CC1(C)C(C)(C)C1(F)C(N1CCCC(NC(c2coc(C3CC3)n2)=O)CC1)=O c1(SCC)cnc(O)c(C(=O)NCC2CC3CC3N2C(C2(OC)CCSC2)=O)c1 C1(NC(CC(=C)C)=O)CCN(C2CCN(C(c3cnc(C(C)C)[nH]3)=O)CC2)CC1 Cc1cc(C)c2[nH]c(=NC3CC(F)(CNC(C4CC5CCC4C5)=O)C3)sc2c1 N1(c2snc(C)n2)CC2CC(NC(c3ccc(CC=C(C)C)cc3)=O)C2C1 c1(C(=O)NC2CN(C(C3C(C)(C)OCCO3)=O)CC(O)C2)onc2c1CCCC2 C1(C(=O)NC(C)CCNC(=O)CC2(C(F)F)CC2)CCOCC12CCCC2 CCC(CNC(=O)Cn1cc2ccccc2n1)N=c1[nH]nc(C(C)(C)C)s1 CCCC(C(=O)NC1CC(NC(C2(C3CCCO3)CCC2)=O)C1)NC(N)=O C1(NC(c2c(OCC)oc(C)n2)=O)CC(F)CN(C(=O)Cc2c(C)noc2F)C1 C1(C)(C(=O)NCC(=C)CCNC(C2CSCN2C(=O)CC)=O)CCSCC1 C1(C(=O)NCCN(C(=O)Cc2csc(Br)n2)CC)CC(=O)NC(C)C1 C1(NC(=O)NCc2c(C)nn(-c3ccc(F)cc3)c2C)CCCCCCC1C C1(NC(c2ccn(C3CC3(F)F)n2)=O)CC(O)(CNC(C2CC2(Cl)Cl)=O)C1 c1(N2C(C)CC(NC(=O)Cc3ccccc3)CC2)ncc([N+](=O)[O-])cc1Br C#Cc1ccc(C(N2CCSCC2C(=O)NC(c2nn[nH]n2)C)=O)c(C)c1 CC(C)C(F)(F)CC(=O)NCCN(C(C1CCC2(C1)CC2(F)F)=O)C1CC1 c1(C(N2C(C)CCC(NC(=O)C(C)(F)F)C2)=O)cnc2cccnc2c1 Cc1ccc(F)cc1NC(C1(C2CC2)CN(C(=O)CNc2ccccn2)C1)=O C1(C(N2CC(C)(C)OCC2CNC(C2(C)COC2)=O)=O)CNC(=O)CC12CCC2 CCC(COC)C(=O)NC(CC)C(=O)NCCC(F)(F)Cl N1(C(c2cn(CC=C)nn2)=O)CC2CN(C(C3CCOCC3)=O)C2C1 N1(Cc2onc(CCC(=O)NC)n2)C(=O)c2ccc(C)cc2C1=O Cc1nc(NC2CCN(C(C3(O)CCSC3)=O)CC2C)ncc1Br C1(C(=O)NC2(CCNC(c3cccc(O)c3F)=O)CC2)CC12CCCOC2 c1(C(N2CC3(C2)C(=O)N3)=O)cnc2n1CCCC2.C1(CC(=O)OC)CC(OC)C1 c1(N(CCN(C)C(c2ccc(CO)nc2)=O)C)nc(Cl)nc2[nH]c(C(C)(F)F)nc12 c1(C(N(C2CN(C(C3C(OC)CCCC3)=O)C2)C)=O)ccc(F)c(C(F)F)c1 c1(C(=O)NC(C)CCCNC(=O)C(O)CC2CCOCC2)ccsc1S(N)(=O)=O c1(C(N2CCN(C(CSC(C)C)=O)CC2)=O)cc2n(n1)CCO2 C=CCCCCC(=O)N(CC(C)NC(c1cnn(C)c1CC)=O)CC c1(C(=O)NCC2N(C(C(CC)C#N)=O)CCC2)cc(Cl)cc2ccncc12 C1(CNC(C2CC(OC)C2)=O)CC(NC(C2(C)CCNC2=O)=O)C(O)C1 c1(C(N2C(C)COCC(COC)C2)C2CCNCCC2)cccc2ccccc12 C1(C(=O)NC2CN(C(c3c(C)nsc3)=O)C(CO)C2)CN2CCCN1CC2 CC1(C(=O)NCCCC2C=NNC2=O)CCN(C(=O)C(c2ccccc2)O)CC1 N1(C(c2cnc(CNC(c3c(C)scn3)=O)nc2)=O)CC2CN(C)CC2(C)C1 c1(CN2C(C(=O)NC(c3ncccn3)CC)CCC2)cc(Br)c(F)cc1F c1(C(=O)NC(c2c[nH]nc2CCCC2CCCN(C)C2)=O)cccc(F)c1F C1(C(N(CC(C)CNC(C2CCC(=O)N2)=O)C)=O)CCC2(CCC2)C1 c1(C(C(=O)NC(CC)Cc2ccccc2Br)(F)F)cccc(F)c1F Cc1c(F)ccc(Br)c1C(=O)NC1CN(C(c2sc(F)cc2Cl)=O)C1 C(=O)(C#CC1CCOC1)N1CC(C(=O)NCCC(C)(C)F)N=CC1 C(=O)(C1=C(Cl)CCC1)NCCN(C(CC=C(C)C)=O)C1CC1 c1(C(=O)NCC2N(C(CC(=O)NCC)=O)CCN(C)C2)cc2ccc(C)cc2[nH]1 c1(CNC(C(COCC)C)=O)ccccc1CNC(c1ccc(COC)cc1)=O c1(C(=O)NCC(C)OCC=C)cc(CNC(=O)C(F)CC2CCC2)nn1C c1(NC(=O)CNC(=O)C(F)(F)F)cccnc1C(=O)NCCN(C1CC1)CC C1(C(=O)NCC2C(NC(=O)CCSCc3ccccc3)C2)CCCCS1 N1(C(C(CCC=C)(F)F)=O)CC(C2CCCN(C(=O)CC3COCCO3)C2)C1 Cc1nn(CC(=O)NCC2C3CN(C(=O)CCOC4CC4)CC23)c(C)c1C CCC(CCOC)C(=O)N1CCOC(CCNC(C2(CO)CC2)=O)C1 C1(NC(CC2(C=C)CN(C(c3nc(Cl)oc3C)=O)C2)=O)CCCC(C2CC2)C1 c1(C(=O)NC2(C)CCN(C(C3(C)CC(C#N)C3)=O)C2)cccc(Cl)c1Cl C(CCCCCN=[N+]=[N-])NC(C1(F)CN(C(C2CCC(N=[N+]=[N-])C2)=O)C1)=O C(=O)(C(C)(C)CCOC)N(C)Cc1cccc(CNC(c2c(CC)scc2)=O)c1 N1(C(C=CCCC)=O)CC(NC(c2scc(C)c2C)=O)CC(F)(F)C1 c1(OC)ccc(CC(=O)NCC2(F)CC(NC(=O)C3CC3)C2)nc1 n1(CC)cc(C(c2nnnn2CC2CCC2)NCC(F)C2CCC2)ccc1=O C1(CNC(c2cccc(NC(C)=O)c2)=O)CN(C(C2OCC2(C)C)=O)CCCO1 c1(C(N2CC3C4N(C(C(C)O)=O)CC(CC4)C3C2)=O)cc2cc(Br)cc(F)c2o1 c1(CNC2CC(NC(c3cc[nH]n3)=O)C2)ccc(I)cc1O C1(C(N2C(CNC(C3(OC)CC3)=O)CC3CC32)=O)CCc2nccn2C1 C1(F)(CNC(Cn2ncc(C)c2)=O)CCN(C(c2ccc(Br)cc2)=O)CC1 Cc1ccc2[nH]cc(CC(=O)NCC(C)CN(C(=O)C(F)(F)C(C)(C)O)C)c2c1 C1(NC2CC(c3ccc(F)cc3)C2)CCCCCC12CCCC2 c1(CNC(N(C(CC)CO)C)=O)cn(-c2ccc(Cl)cc2)nc1C C1(c2cc(CC)no2)CCCCN1C(c1nnc(-c2cccc(Cl)c2)s1)=O C1(C(N(C)CC2CCCN(C(c3c(C)nc(CC)o3)=O)C2)=O)CCC2CCC1O2 c1(NCCSCC(O)Cc2ccc(Cl)cc2)cccc(Br)c1 c1(CN2C(CN(CCCCOCCC)CC(=O)OC)CCC2)ccc(Cl)cc1 CN1CCN(C(=O)COCCNC(c2cn(C)c(=O)n2C)=O)CC1=O C1(C(=O)NCCCN(C)C(c2sccc2Cl)=O)CC(C)(C)CO1 C1(CN(C)C(c2cc(C(N)=O)co2)=O)CCCCN1C(=O)CNS(C)(=O)=O C1(N(C)C(c2cc(Cl)nn2C)=O)CCCCC1NC(c1cnc(C2CC2)o1)=O c1(C(=O)NCC(CCOC)NC(c2cc(C)n(CCO)n2)=O)ccccc1Cl c1(C(N2C(CNC(C(COC)(C)OC)=O)CC2)=O)ccccc1P(C)(C)=O N1(C(CNC(=O)NC)=O)CCCCC1CN(C)C(C1CC1F)=O N1(CCCC)CCCCC1C(N1CCC(CC(C)NC(=O)C(C)C)CC1)=O c1(C(N2CCCC(c3cnco3)C2)C(=O)NCC2CCOC2)cc(F)cc(Cl)c1 N1(C(c2n(CC#N)ncc2)=O)CCCC(NC(=O)CC(F)F)C1 c1(N2C(C(=O)NCc3ccnc(F)c3F)CCC2)ncnc2ccccc12 C(=O)(CC1=CCCC1)NCCN(C(=O)C=Cc1cnccn1)C(C)C c1(OC)cscc1S(=O)(=O)CC.N12CC=CC1NC(=O)NCC1(COCC)CC1C2=O.C(C)C C(=O)(C(CC(C)C)NC(=O)C(CO)NC(=O)C(C)C)NC(c1ncn(C)n1)C C(c1ccc2ncccc2c1)=CC(=O)NC1CC(C)(NC(C(COCC)C)=O)C1 C(CNC(c1ccn(CC(F)F)n1)=O)(CC=C)NC(C(C)OCC#C)=O N1(C(c2n(C(C)C)nnc2)=O)CCn2ncc(CNC(C3CCCOC3)=O)c2C1 CCCCC(C)(C)NC(C1(C)C=CCN1C(C12CC(C#N)(C1)C2)=O)=O C1(CC)(CC)CC(C(=O)NC2CC(n3cc(CN4CCOC4=O)nn3)C2)C1 CC(CC(N)=O)C(=O)NC1COCCN(C(c2ccc(C(F)(F)CF)cn2)=O)C1 C(=O)(C1=C(C#N)CCC1)N1C2CC(CNC(Cc3nc(C(C)C)sc3)=O)C1CC2 Cc1cc(NC(C2CN(C(=O)CN3CC(C)(C)C3)CC23CC3)=O)ccc1C#N c1(C(=O)NC(CCOC)CNC(=O)CC2CC(C(F)F)C2)cc(Cl)cc(F)c1F C(=O)(C(F)(F)C(F)F)NCC(CC)NC(c1cc(Cl)ncc1N)=O N1(C(c2c(CC)non2)=O)CCC2C(NC(C3(C)C=CCCC3)=O)C2C1 Cc1nc[nH]c(=NCC2CN(C(=O)C=CCF)CCC2C(F)(F)F)c1C#N C=C(F)C1(CC(=O)N(C2(C(=O)NCCCCCC)CC2)C)CCC1 C(=O)(C#CC(C)C)N(C(=O)C(C)CNC(C)=O)C1CC(Cc2ccccc2)C1 c1(N2CCC(C(N3CC=CC(NC(=O)CCF)C3)=O)C2)ccc([N+](=O)[O-])cc1 C1(CNC(CCC2(NC(C=CCN(C)CC)=O)CCC2)=O)CCN(C)CC1 C1(C(=O)NC(C)CCNC(=O)C(F)C(F)(F)F)CC2COCC(C1)C2(F)F C1(O)(Cc2ccc(N3CCC(C)C3)cc2)CCCN(C(=O)C2CC2C2CCCO2)C1 N1(C(c2ccc(C)cc2C)=O)CCC2(CCN(C(c3ccnnc3)=O)CC2)C1=O c1(C(=O)NCC(CN(C(c2cncc(CC)c2)=O)C)O)cc(C(N)=O)ccc1C C(CCF)(C(=O)N1CC(C(=O)NC)C1)NC(Cc1onc(CC)n1)=O C(CN=c1c(C)c[nH]cc1C)n1cc(C(c2cc3n(n2)CCC3)CCC)nn1 N1(C(CC(=O)OC)=O)CCCC(C2CCCCN2C(c2ccnc(Cl)c2)=O)C1 N1(C(CCc2ccc(C)s2)=O)CC2CC1CN2C(C1CCCC12CC2)=O C1(NC(CCSC)=O)CN(C(C2CC3C(C2)C3(C)C)=O)CC12CC2 c12cccc(c1)NC(=O)CN1CCC(C1)S2.N(C(C)=O)(CC)CC C1(CN2CCC(C(N(c3nc(Cl)c(-c4ccccc4)s3)C)=O)C2)CCCCN1C C1(CN(C(C)CCC(=O)N(C)C)C(N)=O)CC2(CCC2)CN1c1ccc(C#N)nc1 c1(CC)nc(C(=O)NC2CCC(NC(=O)CN(C)C(=O)OC)C2)c(N)s1 C(CC(=O)NCC1C=CCN1C(c1ccc(O)nn1)=O)(C(F)(F)F)OC N1(C(C2C3(CCN(C(c4cccc(CO)n4)=O)C3)C2)=O)CC2CCOC(=O)C2C1 N1(C(C2CC(NC(C3(C(F)(F)F)CC3)=O)C2)=O)CCc2ccsc2C1 C1(NC(CCNC(CN(C(C)=O)C)=O)=O)CC(CN(CC(F)(F)F)C)C12CCC2 C(=O)(C#CC1CCC1)NCC(CCCC)NC(=O)CC(O)C1CC1 C1(CNCC(=O)N(CC(=O)NC2(CO)CC(OC)C2)C)CCNC(=O)C1 C(=O)(C1(C)CCOc2ccccc21)N1C2C(NC(CC3(NC(C)=O)CC3)=O)C(C2)C1 C(=O)(C=C(Cl)Cl)N(CCN(C(=O)C(c1ccccc1)n1cccn1)C(C)C)C c1(C(=O)NC2CC(NCc3ccc(C)[nH]3)C2)cc(Cl)c(C)c(Cl)c1 c1(CN(S(CC)(=O)=O)Cc2nc(C(=O)OC)n[nH]2)cc(OC)c(OC)cc1[N+](=O)[O-] N1(C(C(=O)Nc2ccc(Br)nc2)=O)CCCC12CCOC2 CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCN(C(=O)C(c2ccn(C)n2)C)C1 C1(NC(c2onc3ccccc23)=O)CC12CCN(Cc1ccc(F)cc1F)CC2 c1(C(N2C(C(N3CC(C)(CCO)C3)=O)C=CC2)=O)ccncc1F CC(C)C(C(=O)N1CC(C)(NC(c2cc(C3CC3)n(C)n2)=O)C1)n1ccnc1 Cc1nnc2n1C(C(=O)NCC1(NC(=O)OC(C)(C)C)CC1(C)C)CC2 Cc1ccc(OC2CCCCC2)cc1CN(C=O)CC=Cc1ccoc1 CCN(OC)C(=O)CNC1C(C)CCC1C C(=O)(CCC(=O)NCCCC1CCN(C(=O)CN(C)C(=O)OC)CC1)NCC C(C1CCCCCC1)=CC(=O)N(C1CCN(C(C2CCN(C)S2(=O)=O)=O)C1)CC n1(CC(=O)NC(CCNC(C=CC(CC)=CC)=O)C)cnc([N+](=O)[O-])c1 c1(-c2nc(C)sc2)cc(C(=O)N(CC(=O)O)Cc2cn(CC(=O)O)nn2)n(C)c1 C1(C(=O)NCC2CCS2(=O)=O)CC12CC(NC(c1cnc(Cl)s1)=O)C2 N1(C(C(=O)NCC)C2COC2)CCN2C(=O)C(C)CC2C1.C1(=O)CCO1 CC(CC(=O)N1CCC1C(F)F)C1CC1 C1(CC)(CNC(C2OCCC2NC(=O)CCCOC)=O)CCC(=O)N1 N1(C(CC(CN(C)C)O)=O)CCC2(C1)CN(C(c1ccc3cnoc3c1)=O)C2 C12(CNC(c3c(CCC)nns3)=O)CCC(CC1NC(=O)Cc1nonc1C)C2 c1(C(N(C2CN(C(C(CC#C)(C)C)=O)CC2O)C)=O)occ2c1CCOC2 c1(C(=O)NC(CC)CNC(=O)C(C)(CO)OC)cc(=O)c2ccccc2o1 CCC(O)CC(=O)NCCn1cnc(C(=O)NC2CC(C(F)F)C2)c1 C(CCCCC(=O)NC1CC2(C1)CC2NC(c1cc(C2CC2)n(C)n1)=O)=CC c1(C(C)C)ncc(Br)c(=NC2CC(NC(c3cccc(F)n3)=O)C2(C)C)[nH]1 CCCC(CCCO)C(=O)N(C1CCC(NC(=O)CC(CC)CCC)CC1)C C12(CNC(CN3C(C)CC3)=O)CC(NC(=O)Cc3ccn(C(F)F)n3)(C1)C2 CCCCCCC(CC)C(=O)NC(C1(CNC(c2cc[nH]c2)=O)CC1)C Cc1cc(=NCCOCC2(CF)CC2)[nH]c(=NCc2cc(C3CC3)on2)[nH]1 C1(N(CCCc2ccncn2)C(=O)OC(C)(C)C)CCCC12CCNCC2 CCC(C)(C)CC(=O)N1CC(N2CCN(C(c3ccon3)=O)CC2)C1 N1(C=O)CC(C)(NC(=O)CNC(N)=O)C1.C1(C(C)=O)(N)CN(C(=O)C2CC2)C1 CC(CC(=O)NC12CCN(C(=O)CCOc3ccccc3)CCC1C2)C(F)(F)F C(=O)(C(F)F)NCCS.C(=O)(CCOCCN)C(C1CC1(F)Cl)=O.C1CO1 c1(OC)cc(N(C(c2ccccc2I)C(=O)NCC2CCCO2)C)c(F)cc1Cl C(CC(C)(C)CC(=O)NCc1ccc(CNC(=O)C=CCCC(C)C)cc1)OC c1(OC)cc(CCC(=O)NC2CC(NC(c3occc3F)=O)C2)ccc1F c1(N2CCC(C)(NC)C2)ncnc2c(Br)cc(C)cc12 c1(C(=O)NCC2C(NC(CN(C(C(C)C)=O)C)=O)CCC2)nc(C(F)F)cs1 N1(C(CCOC(C)C)=O)CCC2CC(NC(c3c[nH]c(=O)cn3)=O)CCC2C1 N1(C(c2n(C)nnc2CNC(=O)C(O)c2ccsc2)=O)CCCCC(CO)C1 Cc1ccccc1C(=O)N1C2(COC2)OC(=O)C1.c1(SCC)ccccc1 C1(CC)CN(C(C2CCN(C3CC3)C2=O)=O)CCN1C(=O)CN1CC2CC2C1 c1(C(=O)NCCC(=O)N(CCCNC(c2n[nH]cc2Cl)=O)CC)ccccc1Cl C1(CNC(C(CC)OC)=O)CN(C(c2cc(C)sn2)=O)CCCO1 C(C)(C(C)C(=O)NOCCCN(CC)CC)NC(C(CCC)CC)=O CCCC(C(=O)NC1(CF)CCN(C(c2cc(C)nc(O)n2)=O)C1)C(C)C c1(C(=O)NC(C(CCC)C)C)n[nH]c2c1CN(C(=O)CCC1CC1C)C2 CC(C)(CF)C(=O)NCC(C1CC1)NC(c1cccc(-n2cccc2)c1)=O C1(C(=O)NCc2c(OC)nsc2)CCc2cnn(C)c2C1.N12CC3(CCC1C3)C2=O C1(CNC(C(CCC)OC)=O)CN(C(c2cccc(C)c2Cl)=O)C(C)(C)C1 CC1CCCN1CCN1CC(CCNC(=O)COC(C)(C)C)C1 N1(C(COC(CC)C)=O)CC2(C(=O)NC3CC=CCC3)CCC1CC2 Cc1cc2c(CC(N3C(CNC(=O)C(C)(C)CF)CC4CC34)=O)csc2s1 C(=O)(CC(C)C(C)(C)NC(=O)C(=O)N(C)C)N1CC2(CC(OC)C2)C1 N1(C(CCC2(NC(C(C(C)C)F)=O)CCCC2)=O)CCC2(CCC(O)C2)C1 c1(C(C(=O)Nc2ccsc2)N(C)Cc2ccccc2)cc(OC(F)F)ccc1F O=C1NCCCCC1C(N1CCCCC1CC(N1CCC(n2ccnc2)C1)=O)=O C(C(=O)NC1CCN(C(=O)COc2ccccc2)CC1O)(C(C)(C)C)N(C)C C1(CC=C(C)C)CCCN(c2ccnc(NC3CCN(C(=O)C(C)C)CC3)n2)CC1 c1(OC)ccc(CN(C)C(c2cc(C)ccc2I)=O)c(Cl)n1 c1(C(N2CCN(C(c3cccc(Br)c3)=O)CC2)=O)onc2c1CNCC2 C(=O)(C(F)(F)c1nccs1)N(C)CC1(NC(=O)CC2(C)CC2F)CC1 C1(NC(C2(CN(C)C)CC2)=O)C2CC3C1C3C2C(=O)NCCF CC(CC(=O)N1CCCCCC1c1ccccc1)(C(=O)O)c1cccnc1 CCC(CNC(=O)CNC(c1ccccc1)=O)(CC)Cc1nn[nH]n1 N1(C(c2ccc(OCC)cc2)=O)C2CCC1CC(NC(C13CCCN(CC1)C3)=O)C2 C1(NC(Cc2c(C)nn(C)c2)=O)CN(C(=O)Cn2cnnn2)CCC1C(F)(F)F CC(C(C)C(=O)N1CCCCC1CNC(c1ccc2nnnn2c1)=O)S(C)(=O)=O c1(C(=O)NC(CCC)C(C)O)cn2c(n1)CN(C(C1CC3C=CC1C3)=O)CC2 C(=O)(C1=CCC(F)(F)CC1)N1CC(C)(NC(c2cc[n+]([O-])cc2)=O)C1 C1(NC(NCC2(OC)CCCC2)=NCc2ccccc2)CC(C)(C)CC(C)(C)C1 c1(C(N(CCCNC(=O)C2=CC(C)(C)C2)C)=O)nc2n(c1Br)CCC2 C1(NC(Cc2c(F)ccc(C)c2)=O)CN(C(C2C(C#N)C2(C)C)=O)CC(F)(F)C1 N1(C(C=CC=CC)=O)CCCC(C(=O)NCC)C1.c1(CC(=O)N)c(C)cnn1C N1(C(CC(=C=C)C)=O)CCC(n2cc(COC(=N)O)nn2)C(O)C1 C1(CC(=O)NCCN(C(C2CC2C(F)(F)F)=O)CC)CCC(C)(C)O1 N1(C(C(C)SC(C)C)=O)CCC(C)(C)C1CNC(=O)C=CC1CCCC1 c1(C(N2CCN(C(C3C(=O)OCC3)=O)C(CF)C2)=O)cn2cnnc2cn1 C1(NC(Cc2ccc(CC)s2)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1F c1(C(N2C(C)CC(NC(C3CC=CC3)=O)CC2)=O)cccc2nc(Cl)cn12 C(C(C)(C)CNC(c1n[nH]cc1Cl)=O)N(C(C(C)NC(=O)OC(C)(C)C)=O)C c1(C(N2CC(O)(C(C)NC(CCC=C(C)C)=O)C2)=O)ncnc(C)c1C N1(C(C2CC2CF)=O)CCC(C)CC1.c1(CC)nc(C(=O)N(C(CCN)CC)C)cs1 N1(C(=O)NC2CCOCC2)CC2CC1CC2CF C1(C(=O)NC2C=CCN(C(=O)CCn3cnnn3)C2)(COC)CCC(=O)N1 c1(C(=O)NCCN2CCCCC2c2n[nH]c(CO)n2)nc2c(cc1Cl)C(=O)OC2 C1(CC(=O)N(C(C)C(=O)NCCCC)C(=O)OCCF)CC2CC2C1 C1(C(CC)(C)C)CCC(C(=O)NCC(O)CCNC(=O)CCC)CC1 c1(C(=O)NC(CC)CN(C(c2ccc(COC)[nH]2)=O)CC)cnc2[nH]ccnc1-2 C1(N=[N+]=[N-])(C(N2CCC(C)(COC)CC2)=O)CCN(C(C2CC=CCC2)=O)C1 N1(C(CN2CCC(C)C2)=O)CCCCC(N(C)C(C2(O)CC2)=O)C1 Cc1ccnnc1C(=O)N(C1CC(NC(=O)C(c2ccn(C)n2)C)C1)C C1(CC)CN(C(=O)C(C)(F)F)CCN1C(=O)CNC(=O)CCCCO c1(C(N2C3C(NC(C(c4c(C)nn(C)c4)C)=O)C(C3)C2)=O)cnn2ccncc12 C(=O)(CCCC(=O)N1CCC(Cn2cc(COC)nn2)C1)NCC c1(OC)cc(C(=O)NCCNC(C23CC(C2)C3)=O)on1.N12CC(C1)C2=O C(=O)(CC(C)C(F)(F)F)NCc1nc(C)c(C(=O)NC(C)(CO)C(C)C)o1 Cc1cc2nn(Cc3ccccc3)c(=O)n2cc1C C(=O)(C1CCCc2ccnn21)NCC1N(C(c2c(CC)nc(C)n2C)=O)CC1 CCC(C(=O)NC1(C)CN(C(=O)C(CN(C)C)NC(C)=O)C1)N(C)C.C(C)(C)(C)SCN c1(C(=O)NC(C(C)C)CNC(=O)CCn2cnnn2)coc2cc(F)ccc12 Cc1nnc(C(N2CC(CNC(=O)CC3CCOCC3)C2)=O)s1 N1(C(C2(C#C)CCCC2)=O)CC(NC(=O)C(C)OCC)C2(CCC2)C1 C12(C(=O)Nc3cc(CN4CCCC4)c[nH]3)CC(C(=O)NCCn3cccn3)(C1)C2 N1(C(=O)OC(C)(C)C)CCC=C(c2cn(C)nn2)CC1.C12CC1OC2=O.C(C)(C)(C)O C(=O)(C#CC1CCCCC1)NC(C1CCN(C(=O)C(C)C2CCC2)CC1)C c1(C(=O)NC(C(C)NC(C(C)C)=O)C(C)C)nccc2c(Cl)cccc12 c1(OC)ccc(C(=O)NC2CN(C(c3ccc(C4CC4)cc3)=O)C2)cc1C CC(C)C(C(=O)N1CC(O)C(N=[N+]=[N-])C1)C(C)NC(C1CCCS1)=O N1(c2c(OC(C)=O)cccc2)CCCN(C(=O)C(F)(F)Sc2ccccn2)CC1 n1(CC(=O)NC2(C(=O)NC(CCOCC)C)CC2)nnnc1C N1(C(CCC(C)(C)NC(=O)Cn2cc(C#N)cn2)=O)CCn2cncc2C1 CCCCC(C)C(=O)NCC(O)CNC(c1cscc1CC)=O N1(C(C2(C)CCCCC2)=O)CC2CCC1C2NC(=O)CC1CCC(=O)NC1 c1(C(c2nnnn2C2CC2)NC(CC=C)C2CC2)ccc2c(c1)CCCO2 Cc1ccc(C(N2CCC(N3CCN(C(=O)C(C)C(C)O)CC3)CC2)=O)nn1 c1(C(N2CCCN(C(=O)C3CC3)CC2)C(=O)NCC(C)C)c2c(nn1C)CCC2 CC1(C(N2CCC(OCCNC(c3ccc(N)c(N)n3)=O)C2)=O)CCC(F)(F)C1 C1(C(N(CC(C)OC)C(C)C)=O)C2CCCC2CN1C(=O)CN1CCCNC1=O C1(COC)(CNC(=O)C(Cl)=CCl)CCCN1C(=O)CS(=O)(=O)N(C)C N1(CCN(C)C(=O)Nc2ccc(C(F)(F)F)cc2)CCC(C(O)C(F)(F)F)CC1 c1(CC)nc(C(=O)NC(C2CCCN2C(c2cc(C3CC3)no2)=O)(C)C)cs1 N1(CC(CCNC(=O)OC(C)(C)C)O)CCC12CC(CC1(NC(=O)O)CC1)C2 C(=O)(C(C)(C1CCC1)NC(c1c[nH]c(C(N)=O)c1)=O)NC(c1ncccn1)CC N(C(=NCCC1CCCN(C)C1)N1CCC2CCCC12)C(CC)CC C(CCCCCC(=O)NCC1CC(C)N(C(c2cncc(O)c2Cl)=O)C1)SC N1(C(CCC(=O)c2ccncc2)=O)CCN(C(C2CCCCO2)=O)C2(CCC2)C1 c1(C(=O)NCC2(OC)CN(C(=O)C(CSC)OC)C2)c(C)nsc1C C(C)(CO)(C(=O)NCC1(CNC(=O)COCC(C)C)CCCC1)OC c1(C(=O)NCC(CNC(c2csc(C)n2)=O)OC)n[nH]c(C)c1Cl C#CC1(C(=O)NC(COC)CO)CCN(C(=O)COC2(C)CCC2)CC1 Nc1cc(C(=O)NCC2CC2CNC(c2cccnc2Cl)=O)c(F)c(F)c1F N1(C(c2n(CC)ccc2)=O)CCCCC(NC(=O)CSCc2cccs2)C1 Cc1ncncc1C(N1CC2C(CNC(C3(C)CC(C)(C)C3)=O)C2C1)=O N1(C(C(C)Oc2ccccn2)=O)C2CCC1(CNC(=O)C(C)N(C)C)CC2 C1(C(=O)NC(CNC(C2C(C)=CCS2)=O)(C)C)CCCCC1P(C)(C)=O C1(CC)(CNC(c2nnnn2CCSC)(C2CC=CC2)C)CCOCC1 N1(c2snc(CC)n2)CCCC(C2CC2NC(c2cc(Br)cnc2NC)=O)C1 Cc1cc2ncc(C(N3CCC(NC(C(F)(F)F)C4CC4)CC3)=O)cn2n1 CCCC(O)C(=O)N1CC2CN(C(c3cnc(O)cc3O)=O)C2C1 C1(NC(=O)Cc2nc3ccccc3[nH]2)CC2CN(C(=O)CC3(O)CCOC3)CC2C1 N1(C(c2c(C)cc(Cl)c(Cl)c2)=O)CCOC2CN(C(c3ccc(=O)oc3)=O)CC12 CC1(C(=O)N2CCC3(C2)CN(C(=O)C=Cc2cscn2)C3)CCc2ccccc21 CCCCC(C(=O)NCC12CC1CN(C(c1ccc(=O)oc1)=O)C2)C(C)C c1(C2(N(C(C=CC)=O)CC)CC2)ccccc1OC.C(=O)C(CC)C1CCOCC1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC2CC(C(N3CC(OC(=N)O)C3)=O)C(C2)C1 Cc1ncnc(C)c1CC(=O)NCC1CC2(CC(NC(C3CC34CC4)=O)C2)C1 N1(C(c2c(C)ncs2)=O)C2CCCC1CN(C(C1CCn3nnnc3C1)=O)C2 Cc1nc(NC(=O)N(CCN2CCCCC2)CC2CCC2)c(-c2ccc(F)cc2)s1 C12(COC(C3CNC(=O)N3)=O)CC(C1)C(C(N1CC(NC(=O)OCC)C1)=O)CO2 c1(C(N2CC(N(C)C(c3cccc(F)c3O)=O)C2)=O)cc(F)cc(S(N)(=O)=O)c1 Cc1ccnnc1C(=O)NCC1CCN(C(=O)CC2CC2(Cl)Cl)C1 c12ccc(cc1C)NC(=O)CO2.C1(C(=O)NC2CN(CF)C2)(COC)CCCC1 c1(C(c2nnnn2C2CCOC2)NCC2=C(C)CCC2)cn2cc(C)ccc2n1 C1(NC(C)(CCI)c2nnnn2CCCC2CC2)CCC2(CC1)CS(=O)(=O)C2 N1(CCn2nnc(C)n2)CCC(NC(C2(C#N)CC(=O)C2)=O)C(C)C1 c1(C(=O)NCCC(C)N(C(=O)CCC2CCN(C)C2)C)c[nH]cc(F)c1=O c1(C(N2CC3C(CNC(C45CC(CC(F)F)(C4)C5)=O)(C3)C2)=O)cccc(F)c1F Cc1cc(C)c2[nH]c(=NCC(C)CNC(=O)CCC3CCC(=O)NC3)sc2c1 Cc1ccccc1C=CC(=O)N(CCCOCCN(C)C(c1cccnc1)=O)C C1(NC(CCN(CC)CC)=O)(CNC(=O)C(C)C(C)(F)F)CCCCC1C O=S1(=O)CCCC(NCc2cnc(C3CC4C=CC3C4)s2)C1 N1(C(C(C2(NC(C(C3CC3)SC)=O)CCC2)C)=O)CCC(CO)CC1 c1(OC)ccc2ccc(C(=O)NC3(c4cccc(Cl)c4)CC3)cc2c1 CCCC(C)(CC)C(=O)NC1CC(CNC(c2ncc(F)cc2F)=O)C1 CC12CCCCC1N(C(c1ccnc(-c3ccco3)c1)=O)CCC2 C1(O)(CCNS(C)(=O)=O)CCN(Cc2cnc(CCN)s2)C1 C(=O)(C#CC(C)(C)O)N(C)CC1CCCC1NC(=O)Cc1cccc(Cl)c1 c1(C(=O)NCC(CC)Nc2cc(C)nn2C(C)(C)C)cc2c(cn1)C(=O)CCC2 C12(C(=O)NCC(=O)OC)C(NC(c3cc[nH]c3)=O)C3CC1C2C3 N1(C(C(C)Oc2ccccn2)=O)CC2(CC(N3CCCC(F)(F)C3)C2)C1 C(=O)(C#CC1(C)CCCO1)NC1CC(CNC(c2cccc(CC)n2)=O)C1 CCC(C)(C)CC(=O)NC(C(=O)N1CCC(n2ccnn2)C1)C(C)(C)O c1(CCC(=O)NCCCCCCCNC(c2cnco2)=O)ccccc1[N+](=O)[O-] C(CCNC(=O)CC1CCCCO1)(C(=O)NCCC12CC(CO1)C2)OC c1(CNC(CCC)CCC)ccc(CO)cc1OC Cc1ccccc1C(C)NC1CC(NC(N2CCC2)=O)C1 N1(C(CC2CC(CC)C2)=O)CCC(NC(c2nc(C)[nH]c2Br)=O)CC1C.N CC(C)CCC(F)C(=O)NCC1(C)COCCN(C(=O)Cc2nc[nH]n2)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2(CC(NC(c3csc(C(F)F)n3)=O)CO2)C1 O=C(C1=CCCOC1)NCc1ccoc1C(=O)NCC1CCC(O)C1 CC(Cc1cnn(C)c1)C(=O)N(CCNC(=O)CCc1ccc[nH]1)C1CC1 CC1C2CCCCC2CN1C(=O)C(CNC(C1CCC(F)(F)C1)=O)CC1CC1 c1(C(CNC(C2(C#N)CCC2)=O)NC(c2ccn(C(F)F)n2)=O)ccc(F)cc1 C#CCC(C)(C(=O)N1CC(C)(C)C1C(=O)OC)NC(=O)CC1C=CCC1 c12ccoc1CC1(CC1)C(C)NC2=O.c1(CC(=O)NCO)cncs1 C(C(=O)NCCCF)(C1=NOC2COCC12)N(c1nn(C)c(CC)c1CC)C N12CC3(CC3C1)C2.c1(N(C)C(=O)C2CC2)ncccc1O.c12ccc(cc1)c(=O)[nH]2 c1(C(N(CCCNC(c2c(CC)con2)=O)C)=O)cc(F)c2ccccc2c1 C(CCCCCCCO)=CC(=O)NC1C(C)CN(C(=O)Cn2nnc(CO)n2)C1 C1(C(=O)NC(CNC(=O)CCN2CCOCC2)C(C)C)(CC)CCCO1 C1(C(=O)NCC(C)(C)CNC(c2ncnc(O)c2F)=O)CC2CCCC(C1)C2 C=C(C)c1ccccc1NC(C1CN(C(=O)CCSC)CC1(F)F)=O c1(C(N2CCC(C)(NC(C(C=C)O)=O)C2)=O)cc2ncc(Br)cn2n1 C(CC(CC)C(=O)N1CCOCC1CNC(=O)CCOc1cccnc1)=CC C1(C(=O)NC(CC)CNC(C23CC(F)C2C3)=O)CCc2cc(OCC)ccc2C1 C(=O)(C(C#N)C(C)(C)C)NC(CC#C)CC(=O)NC1(CC)CCC1 C=CCC(C(=O)NCC(C)(C)C)NC(=O)NCCC1CN(C(=O)CC(C)SC)C1 C(=O)(C1=CS(=O)CCC1)N(C)OCc1c(NC(c2c(Cl)cc(C)s2)=O)cccc1 c1(C(N2CC3(CC3)CC2CO)C(=O)NC(CC)C)cc(C)nnc1C c1(N2CCCC(C)(CNC(C3CC4CCC3O4)=O)C2)ncnc2[nH]cnc12 C1(NC(C=CC(CC)C)=O)CC12CCN(C(=O)CCCc1nncn1C)CC2 N1(C(C(C)n2cnnn2)=O)CCC(C)C(N(C)C(c2ccc(F)c(Cl)c2)=O)C1 N1(C(c2n(C=C)nnc2)=O)CCC(NC(c2cnc(C(F)(F)F)cn2)=O)CC1C N1(C(c2ccc(C(OC)OC)o2)=O)CCN(C(=O)CSC(F)F)C2CCCC12 C(=O)(C(=O)C1=Cc2ccccc2C1)N1C(CNC(c2c(C)cccn2)=O)C=CC1 O=C(C#CC1CCCC1)NC1CC1NC(C1CCCS1(=O)=O)=O C(=O)(C1CC(O)c2ccccc21)Nc1c(C(N(C)C)=O)cc(Cl)nc1 c1(C(=O)NC2CCC(Cn3cc(C(C)OC)nn3)CC2)c(F)ccc2occc12 c1(CC(=O)NCC(CCOC)NC(CCCOCC)=O)ccc(Cl)cc1F c1(-n2cc(CNCCC)nn2)ccc(OC)cc1 c1(C(=O)NC(C2(CNC(C(F)OC)=O)CC2)C)sc2nc(C)cc(C)c2c1C CC(C)CCC(F)C(=O)N1CCCC1C(=O)NC(c1nc[nH]n1)C1CC1 CC(C)C(CC(=O)N1CCOC(CCNC(c2ccncc2F)=O)C1)C(C)C C1(C(=O)Nc2cccc(CNC(CC3(C=C)CC3)=O)c2)CC(C)(C)OC1(C)C c1(OC)ccc(C(N2CC(CNC(C3(F)CCCCCC3)=O)C2)=O)cc1C1CC1 Cn1cnc2c(N3CCCC(CO)C3)nc(N3CC4CCC(C3)N4C)nc12 c1(C(C)=O)ccc2scnc2c1.C1(O)CCCN(C(c2c(C(C)C)n[nH]c2C)=O)C1 N1(C(C(C)NS(CCC)(=O)=O)=O)CCN(C(=O)CN2CCCCC2)C(CCO)C1 S(=O)(=O)(c1cc(Br)c(Br)s1)N1CC2C(C(=O)Nc3ccnc(Br)c3F)(C2)C1 C12(CNC(c3n(CCOC)ncc3)=O)CN(C(=O)C=C3CCCC3)CC1CCO2 CC(C)C(O)CC(=O)N1CC2C(CNC(c3c(N)c(C(F)(F)F)nn3C)=O)C2C1 N1(C(C2C(NC(CC3(OC)CCC3)=O)CCC2)=O)CCCCCC1COC c1(CS(N)(=O)=O)cccc(C(N2CCCC2CCNC(=O)C(O)CC2CC2)=O)c1 N1(C(CCSC)=O)CCC2(CCCN(C(=O)C(C)n3cncn3)C2)C1 c1(C(=O)NCCC2N(C(C(=O)N(C)C)=O)CCC2)nn(C)c2c1CS(=O)(=O)CC2 c1(C(=O)NC2C(C)CN(C(C3CCCC3O)=O)C2)cc(O)nc2c1CCCN2 C=CCC(C(=O)N1CCC(N(C)C)(CC)C1)NC(C1CCCC1)=O N1(C(c2c(CC)nc(C)o2)=O)CCN(c2cc(C)nc(OC)n2)C(CCO)C1 c1(OC)cc(Br)c(NC(=O)CCCc2ccc(Br)c(C)c2)cn1 C(=O)(C(O)C1=CCCCC1)N1CCC(SCC(CN2CCCC(C#N)C2)O)CC1 C=C=C(C)CC(=O)NC(C1(O)CN(C(c2cnn(CC(F)(F)F)c2)=O)C1)C N1(C(c2c(C)onc2)=O)CC2CC2(NC(=O)C(C)C2(O)CCC2)C1 c1(SC)cc(C(=O)NCC(C)(C2CCC2)NC(=O)C(C)Sc2ccccn2)co1 c1(CC)cc(F)ccc1C(N1CCC(CO)(NC(=O)Cc2ccon2)C1)=O c1(C(=O)NC2C(NC(C3CCN(CC(C)C)C3)=O)CCC2)cnn2cnnc2c1 N1(C(CCCOCC)=O)CCC(CO)(NC(=O)C(C)OCCOC)C1 CCC(C(=O)NC1(C)CN(C(C2CC23CN(C(=O)OC(C)(C)C)C3)=O)C1)C(C)(F)F C1(C(=O)NCc2ccccc2)CN(C(=O)C(O)C2CCC2)C2(CCC2)C1 C(=O)(C1=NOC(C)(C)C1)N(CCNC(c1c(C)nsc1C)=O)C1CC1 c1(C(=O)NCC2(O)CN(C(C3C(C)C3c3ccccc3)=O)C2)cc(Cl)ncc1O C12(NC(CN(CC(C)(C)C)C)=O)CCN(C(=O)Cc3cnn(C)c3)CC1C2 c1(CNc2cnn(C3CN(S(C(C)C#N)(=O)=O)C3)c2)nn(C)nc1Br c1(NC(c2cc(-c3ccncc3)[nH]n2)=O)nncn1C1CC1 CCC(C(=O)NCCOC1CN(C(C2(C3CCCCC3)CC2)=O)C1)C(F)(F)F c1(CC(=O)NCCC(C)NC(C2(O)CC2(C)C)=O)nccc2ccccc12 c1(C(=O)NCCC2CN(C(=O)C=Cc3ccccn3)CCO2)cccc(=O)n1O C(=O)(C1=NOC2COCC12)N(C(=O)CC[SH](C12CCC(CC1)C2)CC)CC CCCCC(C)CCC(=O)NC1COCCN(C(=O)CC2CCC(=O)O2)C1 c1(OC(F)F)cc2nn1C2.C1(C)C=CCCC1Cc1ccccc1.CO N1(C(C2CC(OC)C2)=O)CCC(C2CN(C(c3cc(Cl)cc(C)c3N)=O)C2)CC1 c1(C(C(=O)NCC(CO)NC(C(C2CCC2)OC)=O)(C)C)ccccc1C c1(OC)cc(C(=O)NC2CC2CNC(=O)CC2OCCC2(C)C)cc(F)n1 CCC(C)(C(=O)NCC(C(=O)NC1C(=O)OCC1(C)C)N(C)C)C(F)F c1(OC)cnc(C(N2CCC(C(C)NC(=O)CC3CC4CC4C3)CC2)=O)c(F)c1 C(=O)(C(O)C(CCC)NC(C1CC(SC)C1)=O)NC(C#C)(C)C1CCC1 C1(CNC(c2ccoc2)=O)CCCCN1C(=O)CC1CCC(C(F)(F)F)CC1 C=CC1(C(=O)NCCC2CCC(=O)N2)CCN(C(c2occc2C(C)C)=O)C1 C1(C(C)NC(=O)CC2CCCC2)COCC1NC(C12CC(CO1)C2)=O CC1(C)C(C)(C)C1(F)C(N1CCC(C(N2CC3CCCC23)=O)C(O)C1)=O c1(C(N2CCCC(C(C)NC(c3n(CCC)ncc3)=O)C2)=O)cc(C)cc(F)c1 C#Cc1ccc(C(N2CC3CN(C(c4cnc(C(=O)OC)s4)=O)CC23)=O)c(Cl)c1 CC(C)C(C)(O)CNC(=O)COC1CN(C(=O)CCOCC2(F)CC2)C1 Cc1ccc2c(CN3CCC4(CC3)CC4C(=O)O)c(C)ccc2c1 O=C(C1=CCS(=O)(=O)C1)N1CCCCC(CNC(C2(c3ccccc3)CC2)=O)C1 CC(C#N)C(=O)NC1CCC(CNC(c2cc(-c3ccccn3)[nH]n2)=O)C1 c1(CCCNC(=O)NCC2N(CCOC)CC2)c(C)cccc1C c1(CN2C3C(C(=O)NC4CC5(CC(OC)C5)C4)C(C3)C2)c(F)cc(C)cc1F C1(NC(c2cc(C)nn2C)=O)CC=C(C(=O)N2CCCC2CCN(C)C)C1 C1(C(NOC(CC)(CSC)CC)=O)CC2(CC2)CN1C(C1CC=CCC1C)=O C12(C(=O)NCCS(CC)=O)CCCC1CN(C(c1cn[nH]c1)=O)C2 C1(CNC(CC2(OC)CN(C(c3csc(CO)n3)=O)C2)=O)CCC=CCCC1 Cc1cc(N)c(C(=O)NC2(C)CC(NC(c3cc(C)n(CCO)n3)=O)C2)cc1C CN(CCC1CCCCC1)N1CC2(CCN2)CCC1C C=CC(CC)CC(=O)N1CC2CC(C(=O)NC(CO)C(=O)OCC)(C2)C1 C1(F)(CNC(c2c(CC)onc2C)=O)CCCN(C(C2CC=CCC2)=O)C1 C1(NC(C(C)C)=O)CC(CNC(=O)C=Cc2cncnc2O)C12CCC2 CC1(CNC(c2ccnc(Cl)c2N)=O)CCCN(C(c2cc(C3CC3)sn2)=O)C1 c1(NC(C2C(CNC(CC(C)=C(C)C)=O)CCCC2)=O)cncc2ccccc12 C(N=c1[nH]ccnc1F)C1(C)CC(NC(C2CC(O)(c3ccccc3)C2)=O)C1 c1(C(N2CC(C)N(Cc3ccccc3)CC2)=O)cnc2c(c1)OCC(=O)N2 c1(C(N2CCC(N(C(=O)CC3COC(=O)C3)C)C2)=O)ncc2ccccn12 c1(C(=O)NC2CC(CCNC(C3C4CCC(F)(F)C34)=O)C2)ccn2cncc2c1 c1(C(N2CC(OCC)(CNC(=O)Cc3cscn3)C2)=O)c(C)ccc(OC)c1N C(CC1CCCc2ccccc21)(C(CCC(=C)C)C)c1nnnn1C1(N)CC1.OC CS(=O)(=O)c1cccc(C(=O)NCc2ccccc2S(=O)(=O)N2CCCC2)c1F C1(CNC(C(C)CN2CCOCC2)=O)CC2CCC1N2C(C1(C)CCNC1=O)=O C1(C(=O)NCC(CC)NC(c2c(C3CC3)cnn2C)=O)CC=C(C)CC1 C(C(CC(F)(F)F)NC(C12CC(C)(CO1)C2)=O)NC(c1c(C)nccc1)=O CC(CCC(=O)N1CC(CCCCNC(=O)C(C)(O)C2CCC2)C1)N(C)C CC(C)CCCC(C)C(=O)NC1CN(C(=O)CCCC(C)(F)F)CC1C CCC(CC)C(=O)N1CCNC(C(N2CCOC(c3ccccc3)C2)=O)C1 CC(CC(=O)c1cc2sc(n[nH]c1)NCC(C)(CO)NC2=O)CC(C)(C)C C(C(O)CCNC(=O)C(F)c1ccon1)NC(C1(CC)CC1)=O C=CCC(C(=O)NC(=O)CCCn1cc(CSC2CC2)nn1)c1ccccc1 C1(C(N2CC(F)(CNC(C3(C(F)(F)F)CC3)=O)C2)=O)CCC2(CCC2)C1 C#CCCCCC(=O)NC1COCC1NC(c1oc(Br)cc1C)=O Cc1n[nH]c2cc(C(=O)NC3CN(C(C4(C)CC(C)C4)=O)CC34CCC4)ncc12 N1(C(COCCCC(C)C)=O)CCC(NC(C2CCC(=O)N2C2CC2)=O)C(F)C1 C1(C(=O)N(C2CC2C(=O)NCC)Cc2cn(CC=C)nn2)CCN(CCO)CC1 C1(CCNC(C(CC)NC(C)=O)=O)COCCN1C(c1cn(CC)cn1)=O Cc1csc(C(=O)NCCCOCCNC(=O)Cn2cc[n+](C)c2)c1C c1(C(=O)NCC2CCCN(C(c3ccc(C(F)F)nc3)=O)C2)c(O)cccc1Cl c1(NC)cc(-c2cc(Cl)ccc2N)cc(CO)n1 C12(C(=O)NCC3C4CN(C(c5c(Cl)cn(CC)n5)=O)C3C4)CCCC1C2(F)F O=C(C1c2ccccc2CN1Cc1cnc2ccc(Cl)cn12)N1CC(O)C(O)C1 C(C(C)(CO)CN=c1cc(C)nc(N(C(CCO)C(F)F)C)[nH]1)OCC C12(C(=O)NC(CCSC)C)CCCC1CCN2C(c1cc([N+](=O)[O-])c[nH]1)=O N1(C(c2cn(C(C)C)nc2)=O)CCC(O)(C(C)NC(=O)Cc2csc(=N)[nH]2)C1 c1(C(N2CCC(NC(c3cnc(N(C)C)c(Cl)c3)=O)C2)=O)c[nH]c2cccnc12 N1(C(C(C)=CC)=O)CCCC(C2CCN(C(c3ccc(N)cn3)=O)C2)C1 C1(CCNC(c2coc(C3CC3)n2)=O)CN(C(=O)CC2CC2)CCO1 c1(C(=O)NCC2(CN(C)C(c3cnc(N)c(Cl)c3)=O)CC2)n[nH]c2c1CCC2 n1(CC)c2ccccc2c2ccc(CCCCNc3ccc(S(C)=O)cn3)cc12 C1(NC(c2cccc(F)c2)=O)CN(C(=O)C=Cc2cncs2)CC12CC2 N1(C(=O)OC(C)(C)C)CCC12CCCN(C(=O)C(C)(C)ONC(C)=O)C2 Cc1cc(Br)ccc1CCC(=O)NC1CC(C)N(C(=O)CC2CCC2)C1 N1(CC(=O)N(CCN(C(=O)CC2CCCOC2)C)C)CCC(F)(F)C1 C=CCC(C)(C)C(=O)NC1C=CCN(C(c2cc(C)c(C(N)=O)cn2)=O)C1 CC(CC(=O)NC(c1ccccc1)CF)N(C)C(c1nc[nH]n1)=O N1(C(CN(C(C)C)C)=O)CCC(O)C1.C(CC(=O)N(C)CCOC(N)=O)N c1(N(C2CCCCC2)C2CN(C(CC)C(C)C)C2)nn(C)cc1Cl C1(CNC(CCN(S(CC)(=O)=O)C)=O)CCCN1C(=O)C=CC1CCOC1 c1(N(CC(c2ccc(Cl)s2)C)C)cc(NCc2nccn2C(F)F)ncn1 N1(C(CC2(C)CCN2C(=O)COC2CC=CC2)=O)CC(F)CC1CO C1(C2(C)CC2)(C(N2C(C(C)NC(=O)CC3CCCOC3)CCC2)=O)CC1 N1(C(CCCOC)=O)CCC2(CCC(NC(c3nccc(C)n3)=O)C2)C1 N#Cc1ccc(O)c(C(=O)NCC23CCCC(CN2C(=O)C=CCN(C)C)C3)c1 C1(NC(c2ccn(CC)c2C)=O)CCN(C(c2cc[nH]c2)=O)CC12CCC2 C1(NC(C2CC(OC)C2)=O)CN(C(=O)Cc2nocc2C)CC12CCOCC2 N1(CC2CN(C(C)C)C(=O)O2)CCN(Cc2ccccc2)CC1C Nc1c(C(=O)NC2CC(NC(C34COCC3C4)=O)C2)cc(F)c(F)c1F c1(NCC2CC(N3C(=O)CCC3)C2)ccc(S(=O)(=O)NC2COCO2)c(Br)c1 C#Cc1cncc(C(N2CC3CC3(C(=O)NCc3nc(C)co3)C2)=O)c1 C(=O)(C(C)(O)C(F)(F)F)N(C1CCN(CC(N)=O)C1)CC C1(C)(CNC(C(C)=C2CCC2)=O)CN(C(=O)C=Cc2ccncn2)CCO1 C1(CC(=O)NCCC2CC(C)(C)C2)CC2(C1)CN(C(=O)CC1CC1)C2 N1(C(c2ccn(CCC)n2)=O)CC2CN(C(=O)CN(C)C(N)=O)CC2(C)C1 c1(CCC)noc(CCC(=O)NCC(C2CC2)NC(c2coc(Cl)c2)=O)n1 C1(N2S(=O)(=O)CCC2)CCN(N2CCC(N3CCCC3)C2)CC1 N1(C(c2c(C)n(C)nc2)=O)CCC(O)(CN(C(=O)CC2CCCC(=O)N2)C)CC1 C1(N(C(=O)CCCOc2ccccc2)C)CN(C(C2CN(C(C)C)C2)=O)CC1(C)C c1(C(=O)NC2CCCC2NC(=O)C(F)CC2CCCCC2)cnc(C2CC2)nc1 Cc1ccc(C(=O)NC(C)CCCNC(=O)CCC(F)F)cc1OCC(F)F Nc1ccc(C(N2CCC(CF)C2)=O)c(F)c1 N1(C(Cc2c(C)n[nH]c2)=O)CCCC(CCNC(=O)C(c2cccnc2)C)CC1 C1(CCC(=O)NC(C2CC(F)(F)C2)C)CCCN1C(C1CC1(F)F)=O Cc1ncnc(C)c1CC(=O)NCC1CCC(C(N2CC(CC3CC3)C2)=O)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)CCSC)C2)ccc(OC)c(Br)n1 Cc1c(C(N2CC(C)CN(C(C3(C)COC3)=O)CC2C)=O)ccc2c1CCC2 C(=O)(C1CCCc2ccnn21)N1C(CC)CN(C(c2cc(C)cc(C)c2)=O)CC1 c1(C(=O)NCC(N(C)C(C2(C)CCSCC2)=O)C2CC2)cc(=O)cc(Cl)[nH]1 C1(NC(c2c(Cl)cc(C)s2)=O)CCCCCN(C(C2CCCN2S(C)(=O)=O)=O)C1 CCC(C)(COC)C(=O)NC(CCO)CC(C)C.C1(=O)C(C)N1 O=S(=O)(c1ccc(Cl)cc1[N+](=O)[O-])CCn1cc(C2CN3CCN2CC3)nn1 c1(C(=O)NCC(C)C(=O)N(C)Cc2nccn2C)cncc(N(C)C)c1 CCC(COC)C(=O)NC(C1CCCC1)CNC(=O)C(CO)c1ccccc1 c1(C(C)C)cccc(N(C2CCOC2=O)C(C2CCCC2)=O)c1 N1(C(COCCC)=O)CCCC2(CNC(C3CC4(C3)CC(F)(F)C4)=O)CCCC12 c1(CC(Cn2cc(-c3cnc(C(=O)O)s3)nn2)CO)ccc(Br)cc1F N1(C(CCCCOCC)=O)CC2CC1CN2C(=O)CNC(N)=O N1(C(C(CC2CN(C(c3cccc(C)c3)=O)C2)F)=O)CCC2(CC1)CC2C#N C1(NC(C)=O)CCCC(NC(C2(C(=O)NCc3cccc(C(N)=O)c3)CC2)=O)C1 C(=O)(C1=CCCOCC1)NC(C(=O)NC(C(C)C)c1nc[nH]n1)C1CCCO1 C1(CNCc2cn(C)nc2)CC2(CC(NC(c3cc(Cl)ncn3)=O)C2)C1 N1(C(C(C=C)O)=O)CC(=O)NCC1C(=O)N(C)CCN1CCOCC1 O=C(N=c1cco[nH]1)C1CN(Cc2cnc(Cl)nc2)CCS1 N1(C(C(c2c(OC)cccc2)OC)=O)CC(NC(=O)COCCF)CC1(C)C C1(C)(NC(c2cnc(CCC)s2)=O)CCN(C(=O)C(F)=CC2CC2)C1 c1(C(=O)NCCN(C(c2onc(CC)c2C)=O)C(C)C)cnc2n1CCCCC2 C1(n2cccn2)(C(=O)NCCC(=C)CNC(c2cc(Cl)cn2C)=O)CCOCC1 CC1=CCC(C)(C(=O)NC(c2cccc(Cl)c2)CNC(c2ccc[nH]2)=O)CC1 CC1(CNC(=O)CC2C=CCCC2)CCN(CC(=O)NCc2nccs2)C1 C1(C(=O)NCCNC(=O)C(O)C(F)F)(OC)CCCC(C)(C)C1 c1(NC(C2CCN(C(CNC(=O)OC)=O)CC2O)=O)cc(O)c(Cl)cc1Cl c1(CC)cnc(C(=O)NCCCCNC(=O)C(C(C)C)NC(=O)NC)nc1 C12COCCN(C1)C2=O.C1(CC)CC=CCC1NC(=O)CCNC(=O)OC c1(C(=O)OC)ccc(Cl)c(S(=O)(=O)N2CCC3(C2)CN(c2ncc(SC)cn2)C3)c1 CCC(C)CCC(=O)NCC1CCN(C(c2c(C(C)C)cnn2C)=O)C1 N1(C(C(=O)NC(C(=O)OC)C)C2CC2)CCC2(CC(OC)C2)C1 Cc1oc2ncnc(O)c2c1C(N1CC=CC(NC(C2CCO2)=O)C1)=O C1(C(=O)NCC2(C(N)=O)CC2)CC12CCN(C(c1ccsc1)=O)CC2 Cc1nccc(C(=O)NCC(C2CCN(C(C3(N(C)C)CC3)=O)CC2)(C)O)c1N C=CC(C)(C)CC(=O)N1CC2C(NC(=O)C(F)C(C)(F)F)C2C1 Cc1scc(C(N2CC(NC(c3c(C)ncn3C)=O)C2)=O)c1C1CC1 C1(C(=O)NCCCC2N(C(c3n[nH]c(C)c3C)=O)CCCC2)CC(=O)NC(C)C1 C1(CCNC(CC2(N(C)C)CC2)=O)CCCN(C(c2ccc(=N)[nH]c2)=O)C1 N1(C(COCCCC#C)=O)CCC(CO)(NC(c2oc(CC)nc2C)=O)C1 c1(C(=O)NCCCCN(C(C2ON=C(C)C2)=O)C)cn(C)nc1-c1ccc(Cl)s1 c1(OC)ncc(F)c(=NC2CCN(C(c3cc(O)n(CC)n3)=O)CC23CCC3)[nH]1 c1(C(N2CC(C(=O)NCc3nccc(C)c3)C(C)C2)=O)cccn(C)c1=O C1(N(C(CC(C)OC)=O)C)CCCC2CN(C(c3cc(C)nc(O)n3)=O)CC12 CCCC(CC)C(=O)Nc1ccccc1C.c12cn(nn1)CCC1CN(C1)C2=O N1(C(c2c(SC)ccs2)=O)CC2CC2(CNC(C2CCC(=O)N2C)=O)C1 C1(C)(CC)CN(CC)CN1C(=O)C(CC)c1ccccc1 N1(C(C2CC(N(C)C(C3CCCC3)=O)C2)=O)Cc2cc(O)nnc2C1 C1(CCNC(c2cc(Cl)cnn2)=O)CCCCN1C(=O)CC1C=CS(=O)(=O)C1 c1(C(=O)NCCC(CNC(c2c(OC)cccc2)=O)(C)C)cccn(C)c1=O C1(NC(C)=O)CN(C(c2cc3c(nc2C(=O)OC)CCC3)=O)CC12CCOCC2 Cc1ccc(N)c(C(=O)NC(CNC(=O)CC2CC2(C)C)CC(C)C)c1 c1(C(C)(C)C(=O)NC2CC2NC(=O)CC2CC(F)C2)cc(Cl)cc(Cl)c1 c1(-c2cc(Cl)cc(-c3cnc(N4CCOCC4)nc3)c2)cnc2nccn2c1 C(CCCCC(=O)N(C(C)(C)CNC(c1ncc(C(F)F)s1)=O)C)OC C(=O)(CCC(CC)NC(=O)COCC(C)(C)C)NCC1(C=C)CCC1 c1(N2CCN(CCC)CC2)nc(=NCC(O)(CC)CC)[nH]c2c(F)cc(F)cc12 c1(OCCCCNC(c2cn(C)nc2I)C)ncccc1C(F)(F)F c1(C(=O)NC(CC)CNC(=O)CCOCC2CCCO2)ccc(COC)nc1 C1(NC(=O)C=Cc2cc[nH]n2)CC(O)CN(C(=O)CCOCC(F)F)C1 c1(OC)ccc(C(=O)NC(CNC(=O)C(CO)N(C)C)C2CCC2)c2occc12 N1(C(C(C)S(C)(=O)=O)=O)CC2CCCC(NC(c3cc(CO)on3)=O)C2C1 C1(N(C)C)(C(N2CCC(c3cn(Cc4ccccc4)nn3)CC2)=O)CCCOC1 C1(CC(=O)NCC2C=CC(NC(C3N(S(C)(=O)=O)CC3)=O)C2)CCCCC1(F)F CC1=C(C(=O)NC2CC(NC(c3cnoc3C)=O)C2)CCC(C)(C)C1 c1(C(=O)NCC(C2CC2)NC(c2c(C)nsc2C)=O)ccc(Cl)cc1N C(c1cnc(C)s1)=CC(=O)NCC(CC=C)NC(=O)C(Cc1ccccc1)OC C1(F)(CNC(C2CC2(Cl)Cl)=O)CCN(C(c2cncc(-n3cnnn3)c2)=O)CC1 c1(C(=O)NCC2CCCC(NC(C3(C)ON=C(C)C3)=O)C2)ccc(F)c(Cl)n1 C(=O)(C(CN=[N+]=[N-])NC(C1CC(F)(F)C1)=O)NCCC(C(C)C)OC N1(C(C(CC#C)C)=O)CCN(C(C2CC2CC)=O)C(CC(=O)NC)C1 C1(CCN(C)C(C2CC2c2cccnc2)=O)CCN(C(=O)C(F)(F)C2CC2)CC1 C1(NC(C(CC)(C)O)=O)CCCN(S(=O)(=O)c2cn[nH]c2)CC1 c1(C(C)C(=O)NC2CC(CCNC(=O)CC3CC3)C2)ccc2c(c1)OCO2 c1(CNC(C2CN(c3c(OC)cccc3)C2)=O)nc2ncccn2n1 c1(C(=O)NCC2(F)CC(NC(CC=CCC)=O)C2)cc(C)c(C(=O)OC)o1 C1(C(=O)OC)(NC(=O)C(CN(C)C)NC(C2CCOC2)=O)CCOCC1 CC12COC(C(=O)NCCC3CCCCN3C(C3(C)CCNC3=O)=O)(C1)C2 C(CCCC(=O)NC1(C(=O)NOC2CCOC2)CCCC1C)OC C1(CC=C)(NC(=O)COC2CCOCC2)CCN(C(C2(CCN(C)C)CC2)=O)C1 c1(SC(C)C)ncccc1C(=O)NCC1C2CN(C(C3CCCCO3)=O)CC12 c1(CN(C(=O)C=CCN(C)C(C2(C)CCC2)=O)CC)cccnc1 CC(CN=c1[nH]c(=NCCN2CCCOCC2)[nH]c2ccsc12)c1ccncc1 N(C(=NCC1COCc2ccccc21)NC1CCC1)Cc1c2ccccc2sc1 C1(NC(c2c(C)csc2)=O)CCC(C)N(C(=O)COCCC(C)C)C1 c1(C(N2CCC(N(C(C3CC(C)OC3)=O)C)CC2)=O)ccc(S(C)(=O)=O)s1 c1(C(N2CC3C(CNC(C(C(CC)CC)C)=O)C3C2)=O)ccc([Si](C)(C)C)cc1 C1(C(=O)NCc2ncc(C)o2)(CO)CCN(C(C2(c3ccno3)CC2)=O)C1 C1(C)(C(N(CCNC(c2c(OC)c(Cl)sc2)=O)C2CC2)=O)CCCNC1=O C1(CC(=O)NCC2(NC(=O)CN3CCSCC3)CC(F)(F)C2)CCCCC12CC2 C12(NC(C(C)OCCOC)=O)CN(C(c3cnccc3N(C)C)=O)CC1CCO2 N1(C(C23OCC(COC)(C2)C3)=O)CCC(O)C(NC(C2C=CCCC2)=O)C1 C(C(C)C(=O)N1CC(CC(C)NC(=O)CCCc2ccsc2)C1)SC c1(C(=O)OCC2C(C)C2)ccc2c(c1)NC(=O)CCC2 c1(C(N2C(C(=O)NCc3c(C#N)cccc3)CC2)=O)ccc(F)c(Cl)c1F c1(COC)cc[nH]c1C(=O)NCC1CCN(C(=O)CCc2ccn(C)c2)C1 Cc1ccc(SCC(=O)NC(CNC(c2cc(O)ccc2C)=O)CO)cc1C C(=O)(CC1CN(C)c2ccccc21)N(C(CCNC(CCSC)=O)C)C c1(C(N2CCC3(CCC3)C2)C(=O)NCCCCCC)cc(C)c(F)cc1Br n1(C(CC)(C)C)nnnc1C(c1cc(C)co1)NCC1C2COCC12 CCC(CC(=O)NC(CNC(c1csc(Cl)n1)=O)(CC)CC)OC C(=O)(C(C)(O)Cn1cc(-c2cnn(C)c2C(N)=O)nn1)NCC(=O)OC(C)C C1(C(N2CCC(C)C2)=O)CC2CCC1N(Cc1cn(C)cn1)C2 c1(C(=O)NC2CCN(C(CC3C(C)(C)C3)=O)C2(C)C)cc2ccnc(Cl)c2[nH]1 c1(CNCC(N2CC(C(=O)NCC3CCCO3)OCC2)=O)cnc(O)nc1O C1(N(C(CN2C(C)CC2)=O)C)CCN(C(=O)CSc2ccncc2)CC12CC2 CC(CC(=O)NC1CN(C(=O)CC(C(F)F)c2ccccc2)C1)C(F)(F)C(F)(F)F c1(OC)cc(Cl)ccc1CN1CCSCC1C(=O)Nc1cccc(OC)c1C CON(Cc1ccccc1)C(=O)COC(=O)CNC(=O)OC(C)(C)C n1(CC(=O)NC(C(C)NC(CCc2nc(C)c(C)[nH]2)=O)C)cc2ccccc2n1 C1(C(C(=O)N(C(c2ccccc2)CNC(C2(N=[N+]=[N-])CC2)=O)C)O)CCCCCC1 C(=O)(C(CCCCCC)NC(=O)NCc1nccc(OC)c1OC)NC c1(OC)cccc2c(CNC(C)C(c3ccc(F)cc3)O)csc12 N1(C(Cc2scc(CC)n2)=O)CCC(CC)(NC(C2CSCC(=O)N2)=O)CC1 C1(NC(CCOC(C)C)=O)CCCC1(C)N(C)C.C12OCCC1C(=O)N2 C1(C)(CC)CC(NC(=O)CSc2ccc(F)cc2)CN1C(=O)CC=C1CCC1 C(C(CCC)C(=O)NCC(N1CC=CC1)=O)NC(C(C)=CC=C)=O c1(OC)c(C(=O)NCC2CC(NC(=O)C(=O)NC(C)C)CCO2)csc1Cl N1(C(C(COC)C)=O)CC2CC2(NC(c2cnn(-c3cccc(Cl)c3)c2)=O)C1 N1(C(C=Cc2ncc(C)[nH]2)=O)CCCC(C2CN(C(=O)C(C)(C)C(C)(F)F)C2)C1 N1(c2snc(C)n2)CC(NC(=O)Cn2ccc(C)n2)C(C)(C)C1 N1(C(CNC(=O)OC)=O)CC2CCC1C(CNC(c1cnc3scnc3c1)=O)C2 C(=O)(CCC(=O)N1CCC(NC(=O)C(N2CCCC2)C2CC2)CC1)NCCC C1(CC(=O)OC)CN(C(c2c[nH]nc2CF)=O)CC1NC(=O)Cn1ccccc1=O CCC(CC)C(C)C(=O)N1CC2(C(N3CCCC(C(=O)NC)C3)=O)CC1CO2 Cc1cc(CNC(=O)CCOC2CN(C(=O)C(C)(C)C#N)C2)cc(O)n1 c1(NC(=O)NC(C2CC3CCC2C3)C(F)F)cn2ncsc2n1 C(N=c1[nH]c(N(C)CC2CCCO2)nc2c1CCC2)c1cc(OCCC)ncc1 c1(OCC)cc(C(=O)NCC(CCOC)NC(C23CC(O)C2C3)=O)ccc1C N1(C(CNC(=O)NC)=O)CCC2(CC1)CC2C(=O)NCC(C)(O)CC(C)C n1(CC)cnc2nc(=NCC(C)(C)C(C)C)[nH]c(NCCCCCOC(C)C)c12 C(=O)(C1=CCC(NC(=O)CC2(C)CCOC2)C1)NC(CC#C)C(=O)OC c1(C(C)=O)ccc(S(=O)(=O)N(C)C)o1.c12cc(ccn1)C(=O)NCC(C)NC2=O c1(OC)ccc(C(=O)NCC2CN(C(=O)COC3CCOC3)CCC2C)nc1Cl c1(C(=O)NC2CCN(C(=O)CCCc3cccs3)C23CC3)cccc2nsnc12 c1(C(=O)NC(CC=C)CNC(c2ccc(F)s2)=O)ccccc1C1CC1 c1(C(=O)NCCC(=C)CNC(C2(C)CC2C(F)(F)F)=O)cc(Br)cc(C)c1F C#CCCC(O)CCNC(C1(C)C=CCN1C(C1CCOCC1)=O)=O N1(C(C2C(=C)C2C(=O)OC)=O)CCC(OC)(NC(=O)C(CC)OC)C1 O=C1CCC(C(=O)N(CCCNC(C2CCCS2)=O)C2CC2)C1 c1(C(=O)NCC(CNC(=O)CC2CC2)O)oc(C2CC2)nc1C(F)F C1(N(C(=O)CCC2CCCC2)C)CCN(Cc2cncs2)CC1 c1(C(=O)NC(CC(C)NC(C(C)SC)=O)C)oc(S(N)(=O)=O)cc1C c1(C(=O)NCc2c(CNC(CC(C)SC)=O)cccc2)cccc2c1C(C#N)C2 C1(N(C(CCC=C=C)=O)C)CN(C(=O)CCc2cnc(C)s2)CCC1O c1(C(=O)OC)ccc(NCC(C)(C)NC(=O)CN2CCCC2)c([N+](=O)[O-])c1 C(=O)(N=c1[nH]oc2cccnc12)C1(C)CCN1Cc1cnc(Br)c(C(F)(F)F)c1 C(C)(C)(CC(=O)NCC1(C)CSC(C)=N1)NC(C1(CCCC)CCC1)=O c1(OC)ccc(CC(=O)NCC2CCC(NC(c3cc(Cl)on3)=O)C2)c(C)c1 c1(C(=O)NCCCN(c2cncc(Cl)n2)CC)cc(Cl)c(Cl)n1C c1(CNC(c2c(C)cccc2)c2nnnn2C2(C)CC2)cc(F)c(Cl)cc1F C1(CNC(c2ccc(C)c(N)c2)=O)CC2(CN1C(c1sccc1C)=O)CC2(F)F c1(SCCC(N2C(CNC(CCOCC)=O)CC2)=O)ccc(F)c(F)c1 C(c1ccc2c(c1)OCCO2)=CC(N1C(C)CC(NC(C=C(C)C(F)F)=O)C1)=O C#Cc1ccc(C(N2CC3CCCC3(NC(c3c(C)coc3C)=O)C2)=O)cc1F C1(N(C(C23CC(c4ccccc4)C2C3)=O)CCO)CCN(C(=O)CN2CC3CC3C2)C1 Cc1ccc(CC(N2CC(CO)(NC(=O)CNC3CCN(C)CC3)C2)=O)cc1Cl Cc1ccc(-n2cc(C(C)N(C)C(C3CC(F)(F)C3)C)nn2)cc1 C(=O)(C(C)(F)C(=O)N(CCC(=O)OC)CC)NC(COC)C1CC1 N1(C(c2n(CCOC)ccc2)=O)CC=CC(NC(=O)Cc2cnccc2Cl)C1 C1(N2C(=O)c3cc(on3)C2)CC2CC1CN2.C(=O)(C(C)C)OC c1(CC(=O)N(CC2CCN(C(CNC(CC)=O)=O)C2)CC)ccc(F)c(Cl)c1 CC(C)(C(=O)NCC1(F)CCCN(C(C2CCCC3(CC3)C2)=O)C1)C(F)F c1(CC(=O)N(C2CCCN(C(C3(C)CCC3)=O)C2)C)cnn2c1CCCC2 C=CCC(C)(C)CC(=O)N1CC(O)(C(C)NC(=O)CSC2CCOC2=O)C1 CCCC(C)CC(=O)Nc1nc(C(=O)N(c2cccc(C#N)c2)CC)cs1 CN1CC(C(N2CCC(CNC(=O)CCc3nc(O)n[nH]3)C2(C)C)=O)CCC1=O c1(C(N(C(C)CNC(=O)CC2(OC)CC2)CC)=O)c(CC)noc1C C1(NCC(=O)N(C(C)C)C(C)C)CCCCC1N c1(SCC)cnc(O)c(C(N2CCC(CCNC(=O)C(C)(O)C3CCC3)C2)=O)c1 C(=O)(C(CCOCCO)NC(c1cn(C2CCC2O)nn1)=O)OC.C(C)(C)(C)O N1(C(c2ccc(C(=O)OC)o2)=O)CC(NC(C2CCCO2)=O)C2(CCOCC2)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCC12CC1CN(C(=O)C(C)S)C2 N1(C(C2CCCC(F)(F)C2)=O)CCC(CO)=C(F)C1.C12CC(C1)NC(=O)C2 N1(C(C2CC(=O)OC2)=O)CCN(C(c2cnns2)=O)CC1CO Cc1cc(C)c(NC(C2CCCC2NC(=O)CCCN(C)C)=O)c([N+](=O)[O-])c1 C1(c2ccccc2F)(C(N(CC(C)O)CCNC(C(CC)O)=O)=O)CCOCC1 C(CN=C(NCC(F)F)NC1CCOc2ccccc21)(C1CCOCC1)OC c12ccc(s1)NC2.N1(C(C2CC(N3CCCC3)C2)=O)CC(F)(C(=O)O)C1 c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)CCOC)cnc2c(c1)N(C)CCO2 Cc1nc(C)c(C(N2CC3CC3(CNC(=O)CCOCC(F)(F)F)C2)=O)s1 C1(C(=O)NCC2CCCC(CNC(c3ccon3)=O)C2)CCCNS1(=O)=O C(C)(CNC(c1nnn2c1CCC2)=O)(CC(C)C)NC(C(CCC)=CCC)=O C(=O)(C1=C2CCCN=C2NN1)NC1CC(NC(C(CC=C)CC=C)=O)C12CCC2 C#Cc1ccc(C(=O)NCc2ccc(C(=O)NCC(C)(C)N(C)C)cc2)cn1 Cc1cc(=NCCOCC2CC2)[nH]c(NCC(c2cccc3ccccc23)(C)C)n1 Cc1c(CSCCNC(=O)NC2CN(S(=O)(=O)N(C)C)C2)nc2ccccn12 Cc1nc2nccc(N3CCC(F)(CNC(c4cc(C)c(C)nn4)=O)CC3)n2n1 c1(Cn2c(C(=O)Cc3ccnc(-c4ccccc4)n3)ccn2)ccc(Br)nc1Cl c1(C(c2nnnn2C)NC2CC(=C)C2)cnn(C)c1Cl C1(NC(c2cccn2C2CC2)=O)CC2CCC1C(NC(c1coc(O)n1)=O)C2 c1(NC(C)=O)cccc(C(N2CCOC(CN(C)C(C3OCC3(C)C)=O)C2)=O)c1 C(=O)(C1CCc2c(Cl)cccc21)NCC(C)N(C(c1nccn1C)=O)CC Cc1cc(O)ncc1C(=O)NC1CCCCC1CNC(=O)Cc1cc[nH]c1 N1(C(C2(CC=C)CN(C(=O)COC)C2)=O)CCC(C(=O)NCCSC)CC1 c1(C(N2CCOCC(NC(C(C3CCC3)OC)=O)C2)=O)c[nH]c2cc(C)ccc12 c1(C(N2CCN(C(C(=Cc3cccnc3)C)=O)C(C)C2)=O)cccc2sccc12 N1(C(C(CC)n2cncn2)=O)CC(NC(c2cccnc2C)=O)CC1C N1(C(CC2C(NC(CNC(C)=O)=O)CCC2)=O)CCC12CCC(O)CC2 CC(C)C(C)(CNC(=O)CC1CC=CCC1)NC(=O)CCN(CCO)CCO N1(C(c2c(C)onc2O)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1[N+](=O)[O-] c1(C(=O)NCC2N(C(CN(C)CC)=O)CC(O)C2)cc(OC(C)C)ccc1F c1(OC)nccnc1C(N1CCC(C(C)C(=O)NCc2nc(C)cs2)C1)=O C1(CC(=O)NC2CN(C(N)=O)C2)C2CCCC2N1C(C1CC12CCOC2)=O c1(C(=O)NCC(CNC(C(C)CN(C)C)=O)C(F)(F)F)c(Cl)ccc(Cl)c1O CC1CN(C(c2nccn3nnnc23)=O)CC(C)N(Cc2ccccc2)C1 CC1CN(C(=NCCC2CC3C=CC2C3)NC2CC2)CCC1O C(=O)(C(C)(C)CS(N)(=O)=O)NCC(N(C)C(C1(C)CC1C(F)(F)F)=O)C1CC1 C1(C(N2CC(N(C(=O)CCC3CC3)C)C2)=O)CC1C1CCCC1 N1(C(CCCOCC)=O)CC(NC(C2CCC(C)C2)=O)C2(CCS(=O)(=O)CC2)C1 c1(C(N2CCC(CNC(C(C(C)C)O)=O)C2)=O)ccc2c(c1)NCCC(=O)N2 Cn1nnc2ccc(C(N3CCN(C(=O)CCCC4CCC4)C(CO)C3)=O)nc12 n1(CCC)cc(C(=O)NC(C)C(C)(C)NC(=O)C(C)CN(C)C)nn1 N1(C(C(C(=O)OC)(C)F)=O)CCC(C2CCN(C(c3oc(C)nc3C)=O)CC2)C1 c1(NC(=O)NCc2nc(CC)sc2)ccc(OC(F)(F)F)c(NC)c1 N1(C(CN(C)C=O)=O)CCC(c2cc[nH]n2)C1.C1(C(=O)NC)CN(C(=O)C2CC2)C1 c1(C(=O)NCCCCCN(C(=O)CC2CCCCC2)C)c(F)cc(Cl)cc1F N1(C(CCC(C)C)=O)CC2(CCOCC2)CC1CNC(=O)CCC(C)N(C)C CC1(CNC(C2CC3CCC3C2)=O)CCCN1C(c1cnc(C#N)s1)=O CC(C)C(O)C(=O)NCC=CCNC(=O)CSc1nncs1 N1(C(C2C(c3ccn(C)n3)C2)=O)CC2(CCC2NC(c2cc(=O)cc[nH]2)=O)C1 Cc1ccc(NC(=O)C(C2CCOC2)NC(=O)C(C2CCC(=O)N2)C)cc1C N1(C(c2nc(C)sc2)=O)CC(CNC(=O)CN2CC3CCC2C3)CC1(C)C C(=O)(CCN=C(NCc1nc(C2CC2)nn1C)NCC1CCOC1)NC c1(CCC)nc(C)c(C(=O)NC(C2(O)CN(C(c3cc(C4CC4)no3)=O)C2)C)s1 Cc1ccc(SCCC(=O)NC2CCC(C)N(C(=O)C3=CC(C)(C)C3)C2)cc1C C1(N(C)C)CCC(N=c2cccc(S(=O)(=O)NCC(C3(N(C)C)CCC3)O)[nH]2)C1 Cc1c(CN2CCOCC2C)ccc(-c2ccc(C3(C(F)(F)F)N=N3)cc2)c1F c1(NC(c2c(SC(C)C)cccc2)=O)cnc2ccc(Cl)nn12 C1(C(C(=O)NC2CC2)N(C)CC2C(C)C2)CCC(c2ccccc2)CC1 Cc1c[nH]cc(C(N2CCC(C(CO)NC(C3CCC(C)O3)=O)CC2)=O)c1=O CCCC(C)(C)CC(=O)N1CC(C(=O)NCC2(O)CC=CC2)C2(CC2)C1 C1(CC)CN(C(c2cc(Br)cnc2Cl)=O)CC(C)S1=O C1(CNC(=O)CNC(=O)C(F)(F)F)CCCC2(CN(C(=O)C(F)C3CCC3)C2)O1 c1(C(N2CC=C(CCNC(=O)Cc3cccnc3)CC2)=O)ccc2nsnc2c1 C1(C(=O)NCC2(O)CN(C(C(C)O)=O)C2)CN2CCN1CC2C c1(C(N(CCNC(c2c(COC)cccn2)=O)C2CC2)=O)cccc2oncc12 C1(NC(C(C)=C(C)C)=O)CC2CN(C(=O)C=Cc3ccc(F)cc3F)CC2C1 c1(COC)ccnc(C(N2CCCC(C(=O)NCC34CCC(CO3)C4)C2)=O)c1 C(C(C(C)(C)C)NC(C1CCC(CN(C)C)C1)=O)N(C)C.c1(C(=O)N)sccc1CO N1(C(c2cc(OC)c(F)c(F)c2)=O)CCc2nn(C)c(C(=O)NCCSC)c2C1 c1(C(C(=O)OCC)N(C(c2scnc2C)C(C)C)C)ccc(OCC(C)C)cc1 C(=O)(C(CC)CCCCC)N1C(C(=O)Nc2cn(CCC#C)nc2)CC(F)(F)C1 c1(OC)ccc(CN2CCC2CNC(c2ncccc2C)=O)cn1 C(=O)(C(CC(C)C)C(N)=O)N1CCCC(CCNC(c2c(C)coc2)=O)CC1 C(=O)(C(F)(CNC(=O)C(C)N(C)CCN(C)CC)C(C)C)NCC=C C(C1CCN(C(=O)C=CC2CCCC2)CC1)=CC(=O)N(C(CC)C)C Cc1c(C(=O)NCCOCCNC(=O)C(O)C2CCC2)ccc(Cl)c1Cl Cc1ccc(CC(=O)NCC23CC(CO2)N(c2nc(Cl)c(C#N)s2)C3)c(F)c1F N1(C(C2CC(OC)C2)=O)CCC(CO)(CNC(=O)CCOC2CC2)CC1 C12(CNC(CCCC=C)=O)CCCN(C(c3cc(F)ccc3F)=O)C1C2 C12C3CC1CN(C3)C(=O)c1cc(ccn1)N2C.C1(NC(COC)=O)CCCC1 C(=O)(CC(F)(F)C(F)(F)F)NCC1(CNC(c2ccc(OC)cc2Cl)=O)CCC1 CN1CC2(C(=O)NCc3ccn4ccccc34)CC(C3CC3)C12 c1(C(C(=O)NC2CC(N(C)C(C3CC3(C)C)=O)C2)(F)F)ccc(F)cc1 N1(C2CN(C(C(C)=C3CCCC3)=O)C2)CC(NC(=O)Cc2sccc2C)CC1=O C(=O)(C1=C(Cl)CCCC1)N(CCNC(=O)CC)CCOCC(=O)NCC1CCC1 C1(CC)CN(C(=O)COC)CC(N(C=O)C(C)C)O1.C(COCCOC)S c1(C(N(CCOC)CCNC(=O)C=Cc2ccc[nH]2)=O)c(SC)cnn1C CC1(C)CC(CC(=O)Nc2ccc(CO)nc2)N(C(C2CC3(CCO2)CC3)=O)C1 [N-]=[N+]=NC1CCC(C(=O)NCc2ccc(CNC(C3CSC3)=O)c(F)c2)C1 C1(O)(C(N2C3CC(NC(C45OC(C)C(C4)C5)=O)C(C3)C2)=O)CN2CCC1CC2 C12(C(=O)NCC3CC3)CCN(C(C3CCC4(CCC4)C3)=O)CCC1C2 c1(C(N2C(CC)CN(C(C3CCCCC3)=O)CC2)=O)nc2sccn2c1C C#CCCCC(C)C(=O)NC(CC1CCC1)C(=O)N1CC(C(C)(C)C)C1 CC1CN(C(=O)NC(C(C)(C)NC2CC2)OC)C1 C(=O)(C#CC1(C)CC1)N(CCN(C(=O)CC1(CO)CCOCC1)C(C)C)C N1(c2c(CCC)cccc2)C(=S)NC(c2ccccc2CC)C(C(=O)OC)=C1C CC(C)C(C(C)C)C(C(=O)NCCCC1CCC1)N1Cc2ccc(Br)cc2C1 CN1CCC(NC)C1=O.C12(CC13CCC3)C(OC)C1CN(C1CO)C(=O)NC2 C12(C(=O)NCC(CC=C)NC(=O)C(c3ccccc3)O)CC(C1)C(C)(C)O2 C(=O)(CCC(=O)NCC(O)CNC(=O)CC(c1cccc(F)c1)C)N(C(C)C)C C1(CC=C)(NC(=O)CCc2cc[nH]n2)CCN(C(=O)CCCN2CCCC2)C1 C(=O)(C(C(=O)NC(c1ccccc1)CNC(C1(OC)CC1)=O)C(C)C)OCC CC1CN(C(C2CC2C2CCC2)=O)CC1NC(=O)CN1C(=O)CCC1=O CC(C)S(=O)(=O)CC(=O)NC12CC1CN(C(c1cocc1Br)=O)C2 CC1(C)CCCC(O)(C(=O)NC2CCC(NC(C3CCN3C(C)(C)C)=O)CC2)C1 c1(CNC2(CCC)CCOC2)ccc(O)c(OC)c1 c1(OC)ccc(C(F)(F)C(=O)NC2CC(NC(c3sccc3Cl)=O)C2)cn1 C(CC(C)CCNC(C1(F)CC1(F)F)=O)NC(c1ccn(CCC)n1)=O C(N=c1[nH]c(N2CCC(CC(F)F)C2)nc2c1CCCCCC2)c1nc(Br)sc1 Cc1cccnc1C(=O)NCCCC1CCCCN1C(=O)CN1CCSCC1 Cc1nc(CCC(=O)NCC(F)(F)CNC(=O)Cn2cncn2)oc1C C#Cc1ccc(C(=O)NC2(C(=O)NCc3ccsc3C)CC2(C)C)cc1C c1(C(=O)NCC(CC(C)C)NC(=O)CCn2cc(Cl)cn2)cc(F)cc(N)c1F c1(CCC)cccc(C(=O)NCCCC(C)NC(=O)C(C)SC(C)C)c1 c1(C(N2CCN(C(C(=O)NCC(C)C)=O)C3C2C3)=O)ccc(S(=O)(=O)N(C)C)cc1 N1(C(=O)OC(C)(C)C)CCC2CC(C(N3CC(O)C4(CCCC4)C3)=O)CCC12 c1(OCC)nc(C(=O)N(C(C)CNC(=O)CNC(c2ccoc2)=O)C)co1 C1(CNC(C(C)N(CC)CC)=O)CC(C)N(C(=O)CN(S(C)(=O)=O)C)C1 CC(C)(C)CC(F)C(=O)N1CCCC1CC(=O)NC1CCCSCC1 C(=O)(C1=CSCCO1)NC(C(C(C)C)NC(c1cn(CCC)nn1)=O)C C1(CC(=O)NCCN(C(C)C)C(C2CCC2(F)F)=O)(N(C)C)CCCC1 c1(C(C(=O)NC(CC(=O)OC)C)(C)OC)ccccc1Cl Cc1ccn(C)c1C(=O)NCC(C)NC(C1COC(=O)N1C)=O C=CCC(CC(C)C)C(=O)NCCCC1CCCCN1C(=O)C#CC(C)(C)C=C C1(NC(C(CC)(F)F)=O)CC2CC1CN(C(c1cnc3nccn3c1)=O)C2 N1(C(CSCC(N)=O)=O)CCC2(CCOCC2)C(NC(c2ccn(C(F)F)n2)=O)C1 N1(Cc2cn(C)nc2)CCC(F)(F)C(NC(c2ccc(Br)cc2Cl)=O)C1 C(=O)(C(CCC1CC1)NC(=O)Cc1ccc(F)cc1)N(CC(C)O)C N1(C(C(=O)Nc2n(CC)c(O)nc2)=O)CCSC(c2ccc(C(C)C)cc2)CC1 N1(C(CCC#CC)=O)C(CC(=O)NCC(c2cnn(C)c2)O)C2CCCC12 C(=O)(C1=NNC(=O)C1)N1CC(OC)(CNC(c2cncnc2C)=O)C1 C1(NC(c2c(OC)ccs2)c2nnnn2Cc2cccs2)CCC(C)(C)CC1C C1(NC(CC(=O)OC)=O)CC(NC(=O)C(C2CCOCC2)C)C12CCOCC2 n1(C(C)C)[nH]c(C(=O)NC2CN(C(=O)C(c3ccc(F)cc3)O)CC2C)cc1=O c1(C(N2CC(OC)CC(NC(C(CC#C)C)=O)C2)=O)ccc(C#N)cc1C C1(C(=O)NCCC2CC(C)C2)CC2C=CC1N(C(=O)Cc1n[nH]c(C)n1)C2 Cc1csc(=O)n1CC(=O)NC(C)CNC(=O)CN1CSCC1=O C(=O)(CCC(=O)NC1CCC(NC(=O)C(C2CCOC2)SC(C)(C)C)CC1)NC N12C3CCC1CN(C3)C(=O)Cc1ccc(s1)C2=O.c1(CC)ccc(OC)cc1Cl N1(C(C(c2ccnn2C)C)=O)CCN(C(c2cc(=O)n(C)cn2)=O)CC(O)C1 C1(CC(=O)NC2(C(N3CCC3C3CCC3)=O)C(C)C2)CCOCC1 N1(C(CC(=O)NCC)=O)CCC(NC(c2ccccc2OCC2CC2)=O)C1C c1(C(=O)NC(CNC(C2C(=C)C2)=O)CC)ccc(C#N)c([N+](=O)[O-])c1 c1(C(=O)NC2C3CCN3C2=O)ncccc1O.C1(COC)CCCC(CF)C1 C(C(C)(C)C(=O)N(C)CCn1cccn1)N(C(C1CC(OC)C1)=O)C N1(CC2NCCN(S(=O)(=O)Cc3ccccc3)C2)CCn2nccc2C1 C1(CC)CCCN1C(=O)C(C)CN1CCOCC1.CCC1CNC(=O)C(=O)N1 C1(C(=O)NCCCC(=O)OC)CC2CC1CN(C(C1CC(C(F)(F)F)C1)=O)C2 C1(C(=O)NCCC(C)NC(C2CCCOC2)=O)CC2(CSC2)C1 c1(C(N2CCN(C(COCCCC)=O)CC2C)=O)cnn2c(C)ccnc12 C1(C(=O)NC(CC(C)C)C)CC2CCCC2N1C(=O)CCC1CCC1 C(c1ccccc1Cl)=CC(=O)NCC(CC(C)C)NC(C1(N(C)C)CC1)=O Cc1cc(C(=O)NC(C)(CNC(c2scnc2C(F)F)=O)C2CCC2)sc1C C(=O)(CC1C(=O)Nc2ccc(F)cc21)NCC1(O)CN(C(C(CC)F)=O)C1 C=C(C)CCC(=O)NCC(C)(C)NC(C1C(c2nc(=N)[nH][nH]2)C1(C)C)=O N1(C(C(c2cccc(Cl)c2)SC)=O)CCC12CN(C(=O)C(F)F)C2 c1(NC(C2C3CN(C(c4csc(Cl)n4)=O)CC23)=O)ccccc1N1CCCC1 C(=O)(C(C)(C)CNC(C1CCC2(CC2)C1)=O)N(CCC)C1CC1 O=[N+]([O-])c1cccc2[nH]cc(CNCc3coc(C(F)F)n3)c12 c1(C(N(C)CC2CCN(C(C(C(C)C)F)=O)C2)=O)cnc2n1CCCC2C N1(CCCS(C(C)(C)C)(=O)=O)CCOC2(CCN(C(c3cncnc3)=O)CC2)C1 c1(CC(=O)NCC2OCCN(C(CC(COC)(C)C)=O)C2)coc2ccccc12 C1(O)(C(C)NC(c2cc(C#N)cs2)=O)CCN(C(c2sccc2F)=O)CC1 c1(CNC(c2c(C)nc(-c3c(C)ccnc3)s2)=O)ccc(C)c(C)c1C C#CCC(CC#C)C(=O)NCC1CC1CNC(=O)CN(S(C)(=O)=O)C N1(C(C(N2CCOCC2)C)=O)CCC2CN(C(c3cc(Cl)ns3)=O)CCC12 C1(NC(C(CC=CC)C)=O)CN(C(c2ccc(=N)[nH]n2)=O)C(C)(C)C1 c1(C(=O)NC2C=CC(CC(=O)N(C)CC3(C)CCCO3)C2)cccc(O)c1F c1(C(=O)NC2CN(C(c3ccc(C(C)=O)o3)=O)C(C)CC2)cc(C)c(C)cc1N N1(C(C2(F)CCOCC2)=O)CCC(CNC(=O)C(F)(F)C(F)F)C(C2CC2)C1 CCC(C#N)(CC)C(=O)NCC1CN(C(c2conc2C(F)(F)F)=O)CC1(F)F O=C1NC(C2CCCOC2)C(=O)N1C(c1ccc(Cl)cc1F)c1ccncc1 C1(C(=O)NCCC2CN(C(C3(Cl)CC3(F)F)=O)CCO2)(OCC)CCSCC1 O=C(CCSCC(F)(F)F)NCC(C1CCCO1)N(C(C1(F)CC1)=O)C1CC1 C#CC1CCN1C(=O)C=CCC(C)(C)NC(c1cccnn1)=O N#Cc1ccc(CNC(=O)CCC2CCC(NC(=O)CC3CCCC(O)C3)C2)o1 CS(=O)(=O)C(C(=O)NC12CC(C1)N(C(=O)CCCC1CC1)C2)C1CC1 C(=O)(C1CCN(C)c2ccccc21)NC(c1ccc(C)cc1)CNC(=O)C(O)CF c1(C(N)=O)nccnc1C(N1CC(F)(C(=O)NCCc2cnccn2)C1)=O Cc1nc(C)n(Cc2ccc(N(C(=O)CSNc3ccccc3C)C)cc2)n1 Cc1nc(C(=O)NCC(C(C)C)NC(=O)C=CC(C)(C)C)n(C)n1 c1(-c2c(C(=O)NC3CN(C(C(CC)O)=O)CC3F)nco2)c(F)cccc1F c1(C(=O)NC2CC3CN(C(CN(C(C)=O)C)=O)C2C3)nnn2c1CCCCC2 c1(NC2(NC(c3ccc(O)nc3)=O)CCC2)ccc2nnnn2n1 C1(CNC(c2cc(CCC)n(C)n2)=O)CC(C)(C)CN1C(=O)CC(O)CCSC c1(C(=O)NCC2C(NC(C3CC(C(F)F)(OC)C3)=O)CC2)ccc(C(F)F)nc1 C(=O)(CC(C)(O)C(F)(F)F)NC1CC(C)(C)N(C(=O)CN2CC3CC3C2)CC1 C(=O)(CCCS(N)(=O)=O)N1CC(C)(C)C(NC(C2CCn3ccnc3C2)=O)C1 Cc1cc(OC(=O)CO)sc1C(N1CC(CNC(c2ccc(Cl)cc2)=O)C1)=O c1(OCC)ccc(-c2nnc(C(C)C)o2)cc1.C1(CN)(CO)CCCOC1 C1(S(=O)(=O)OC(C)(C)C)(C(N2CCC(N(C(C(F)OC)=O)C)CC2)=O)CCC1 c1(C(N2CCCC(N(C)C(C3CC(C(F)F)C3)=O)C2)=O)nccc2ncncc12 c1(NC(C2CCC(NC(c3cccc(F)c3)=O)C2)=O)nc[nH]c2nccc1-2 N1(C(c2cnc(C)[nH]2)=O)CCCC12CCN(C(=O)C(F)CC(C)(C)C)C2 CC1CC(C(N2CC(CNC(=O)CC3(C)CC3(F)F)C2)=O)CO1 C1(NC(C2C(CCC)C2)=O)CCC(NC(c2cc(CC(C)C)nn2C)=O)CC1 c12cccc(c1)OO2.N1(CCCOC)CCC(NC(C)=O)CC1 S(=O)(=O)(c1ccccc1C#N)N1CC(CC(=O)Nc2c(OC)cc(Br)cc2Cl)C1 N1(C(CC2N(C)C(=O)CC2)=O)CCC2(CCCN2c2nc3ncc(Cl)cc3o2)C1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C(C)C2)cc(COC)c(OC)cc1C c1(CN(C(C(C)OCC=C)=O)C)ccccc1CNC(C1(CCC)CC1)=O C(C)(C)(CC(=O)NCC1CCN(C(=O)CCCCc2ccccc2)C1)N(C)C N1(C(COCCC(C)C)=O)CC(CNC(=O)C=Cc2ccoc2)C(C)(C)C1 c1(C(C(=O)NCCOC)N(c2ccccc2Cl)CCC)nnn2c1COCC2 c1(CCNC(C2CC(=O)N2)=O)ccc(N2CCN(C(=O)CS(C)(=O)=O)CC2)cc1 C1(CC=C)(NC(=O)C(C)C(O)CC)CCCN(C(=O)Cc2ccsc2)C1 C(=O)(C(F)CC(C)C)NC(C1N(C(C(n2ccc(C)n2)C)=O)CCC1)C c1(C(N2CC(n3cc(C4CC4)nn3)C(O)C2)=O)cc(F)cc(F)c1.C12CC(C1)O2 c1(C(=O)NCC2OCCN(C(C(CC=CC)C)=O)C2)cnc2c(ccn2C)c1 CN(C)NC(=O)CCC(=O)N1CC(O)(C2CCCN2C(=O)C(C(C)(C)C)N(C)C)C1 N1(C(=O)COCCS(=O)(=O)N2CCCC2)CC2(C1)CN(C(=O)Cn1nccn1)C2 c1(CC(=O)NCC(CN(C(C(C)(CO)OC)=O)C)C)cc(Cl)cc2c1OCC2 C1(n2cc(CC(OC)OC)nn2)CCC(NC(C2CCOC2)=O)CC1 c1(C(C(=O)NCCC2(C)CC2)N(C2CC(F)(F)C2)CCC#C)cc(F)ccn1 C1(CNC(C2(SC)CC2)=O)(CNC(C2(C)C=CCCC2)=O)CCCCC1 C1(C(=O)NC(CCC)C)CCN(C(=O)Cc2cncc(O)c2)C1(C)C n1(CC)nnc(C(N2CCC(N(C(C34CCC3C4)=O)C)CC2)=O)c1N.C(C)(C)(C)S Cc1cc(C)c(CC(=O)NC2C3CC2N(C(=O)C(C)(C)n2cccn2)C3)c(O)n1 C1(O)(CC(N2C(CC(=O)NC(CO)(CO)CO)CCC2)=O)CCCCC1 C(=O)(C1=NNC(=O)CC1)NC1C(CNC(c2nc(OC)oc2)=O)CCC1 Cc1nc(C)c(CNC(=O)CONC(c2c(C)noc2N)=O)o1 N1(C(C(c2cc(=O)cc[nH]2)(C)C)=O)CCC2(CCN(C(=O)CCF)C2)C1 c1(C(N2C3(CNC(C(C)OC)=O)CC(COC)(C2)C3)=O)ccc2[nH]c(=N)[nH]c2c1 CCC(C(=O)NNc1cc(C)c(C(=O)OC)cn1)SC c1(C(c2n(C)nnn2)Nc2cn(C)nc2C#N)ccc2c(c1)CCCO2 c1(CN2CCC(Oc3c(C)cccc3)CC2)ccc2c(c1)nnn2C C1(C2CC2)(C(=O)NCC2CN(C(C3CC3(F)Cl)=O)C2)CCOCC1 c1(C(N(C(C)CNC(c2cncc(Cl)c2Cl)=O)C)=O)cc2n(n1)CCCNC2=O c1(OC)ccc(CN(C(c2ncoc2C)C(=O)NCc2ccco2)C)cn1 CC1(C)CCCN(C(C2CCCCC2O)=O)C1C(=O)NC1CC2CC2C1 c1(CNC(C(COCC)n2ccnc2)=O)cc(C)ccc1OCCOC(C)(C)C N1(C(C2(C#C)CCC2)=O)CCC(N(C(c2ccc(CSC)cc2)=O)CC)CC1 N1(C(COCc2onc(C)n2)=O)CC2CCC1C(NC(C1CC1(Cl)Cl)=O)C2 Cc1cccc(C(O)C(=O)OCCCCC(=O)N2CCN(c3nnc(C)s3)CC2)c1 CC(O)(CC(=O)NC12CCC(C(=O)NCC34CCN(CC3)C4)(CC1)C2)CC(=O)O CC1CC(NC(=O)COc2ccccc2)CCN1C(=O)CC1CCC1 N1(C(c2cc(C)c(CO)cn2)=O)CC2(CCN(C(C3CCCC(O)C3)=O)CC2)C1 C1(C)(C(=O)NC(CN(C)C(C2CCCOC2)=O)(CO)CO)CCCNS1(=O)=O Cc1ccc(C(=O)NCCOCCCN(C)C(C2CCCCS2)=O)c([N+](=O)[O-])c1 C1(CC)(NC(c2ccc(O)c(CO)c2)=O)CCN(C(=O)Cc2ccccn2)CC1 O=C1CCCC(CCCC(=O)N2CC(C3CN(C(C4CC4(F)F)=O)CCO3)C2)N1 c1(-c2c(OC)csc2)ccc2cc(C(=O)Nc3ccnc(OC)c3Br)sc2c1 C1(C(=O)NCCC(C)C)(CNC(C(CC)=CCCC)=O)CC12CCC2 CCCCC(C(=O)NCC1C=CC(NC(=O)C(C)OCC2CCCO2)C1)N(C)C c1(N(C)C)ccccc1Br.n1(C(C2CCC2)N)cc(C(O)O)nn1.C(COCCOC)NC.O C12(CNC(=O)C=CBr)CCC1CCN2C(c1ccc(Cl)cc1)=O C(=O)(CCC(=O)C(C)(C)C)N1CCCC(C(C)NC(=O)CC(C)(C)C)C1 c1(C(N2CCC(C(C)(C)NC(C3OCCN(CC)C3)=O)C2)=O)cc2scnc2[nH]1 N1(CC(=O)NCC(F)(F)F)CCOCCC1CC.c1(C(=O)OCC)sc2nc1-2 N1(C(C2(C)CN(C(C3CC(=O)OC3(C)C)=O)C2)=O)CC2(CCC2(C)C)C1 C1(CNC(C(CC)COC)=O)CCN(C(c2ccnc(O)c2)=O)CC1C C(=O)(CS(=O)(=O)C(C)C)NCCCC1N(C(CCC=C(C)C)=O)CCCC1 C#CCC(CC(F)F)C(=O)NCC1COCCN(C(c2cnc(C(N)=O)s2)=O)C1 C1(C(=O)NCC(C2CCC2)NC(C(C=C)c2ccccc2)=O)CC2(CSC2)C1 Cc1c(C(=O)NCCCCCNC(=O)C2=NNC(=O)C2)ccc(C(F)(F)F)c1F c1(C(=O)NCC(c2cccc(OC)c2)NC(C2CC2F)=O)c(F)ccc(F)c1N C1(C(=O)NC2CCN(C(C3(COC)CC3)=O)C(C)C2)CCC(C2CCCO2)O1 C1(C(N2CC3(CN(C(C)=O)C3)C2)=O)CC2(CCN(C(=O)C(C)OC(C)=O)C2)C1 c1(Cc2nc(CCCOC)nn2-c2ccc(C)c(Cl)c2)ccc2nc[nH]c2c1 Cc1ccc2nc(C(=O)NC3CCCN(C(C4CC(C)(F)C4)=O)C3C)cn2c1 c1(C(=O)NCCOCCNC(Cn2c(C(C)C)nnn2)=O)ncncc1Cl N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC2(CC(NC(=O)CSc3ccncc3)C2)C1 CCC(CCC(=O)N1CCOC(C(=O)NC(C2CCOCC2)(C)C)C1)OC C12CCC3(CCN(CC3)OC(=O)N1CC=CCO)CO2.C(C)(C)(C)NC(C)=O C(C)(C(C(=O)NCC12COC(C1)C(O)C2)C(C)C)NC(c1noc(CC)c1C)=O c1(OC)ccnc(N(C2CNCC2C#N)C(=O)C(C)Nc2ccccc2)n1 C(=O)(C(C)(C)C(=O)NC(CNC(=O)C#CC1CC1)C(C)C(C)C)NC Cc1cc(C(=O)N(C2CCN(C(c3sccc3C)=O)CC2)CCO)[nH]c1C C(=O)(C1(C)CCc2ccc(Br)cc21)N1CC(C2CN(C(C(COC)C)=O)C2)C1 N1(C(C2(CC)CCNC2=O)=O)CCCC(CCNC(c2ccc(C)nc2)=O)CC1 c1(C(N2CC(C)N(C(c3cncs3)=O)CCC2)=O)ccc2c(c1)COCO2 N1(C(C(C)N(C)C)=O)CC2CCC(N(C)C(C3CC4C=CCC(C3)C4)=O)C2C1 C1(CNC(Cc2nc(C)oc2)=O)CN(C(=O)CCN(C2CCCCC2)C)CCO1 CC1CCN(C(c2[nH][nH]c(=N)c2Br)=O)CC1CNC(C1CCC1)=O CC1CN(C(c2cnsn2)=O)CC1CNC(=O)C(C)(C)CF Cc1nn(C)c(C(N2CC(CNC(C3CC3(C)C)=O)C(C)C2)=O)c1Cl C1(C(=O)NCC2(C)CCCCCCC2)CCc2ccccc2C1 c1(C(N(CCCCNC(C2(SC)CCC2)=O)C)=O)ccc(C)c(C(C)=O)c1 C1(CC)C(C(N2CC(N(C(=O)C(C)(C)F)C)C2)=O)CCN1C(=O)OC(C)(C)C Cc1ncc(CNC(c2ccc(CCC(=O)NCCCCO)[nH]2)=O)o1 C(=O)(CCC=CBr)NC(CN(C(=O)C(C)(C)c1ccc(Cl)s1)CC)C CCCCC(C(=O)NC(C)(CC)CCNC(C1CNC(=O)O1)=O)N(C)C CC(C)(C)CCCC(=O)N1CCCCC(CNC(=O)CC(C)(C)C)C1 Cc1cccc(NC(N2CC(n3cc(C(C)C(=O)O)nn3)C(C)C2)=O)c1 c1(C(=O)NCC(CNC(c2cnoc2C)=O)OC)cc2c(F)cc(F)cc2o1 Cc1nn(CC(F)F)cc1C(=O)NC(C)(C)CCNC(C1COC(C)C1)=O N1(C(C(CC)=CC)=O)CCC2CCCC12C(=O)NCC(C)COC C1(C(=O)NC(CNC(C(CC)=CC)=O)C)CC2CC1CC2(F)F N1(C(C(C)OCC#C)=O)CC(NC(=O)COCCOCC)C(c2nccn2C)C1 c1(CC(=O)NCCC2(O)CCN(C(C(CC)COC)=O)C2)c(F)cccc1Cl C(CCC(=O)NC1CC(O)C1CC(N1CC(C)(N(C)C)C1)=O)OCCC N1(C(C2(C)CC(=C)C2)=O)CCC(C2CCN(C(=O)Cc3cccs3)C2)C1 C(CC(C(=O)N1CCCCC1CF)NC(=O)Cc1ccn(C)n1)OC N1(C(C=CC(C)C)=O)CCCC2(C1)CN(C(C1CCCNS1(=O)=O)=O)CCO2 c1(C(=O)NC2C(NC(C3CC(C(F)(F)F)(OC)C3)=O)C2)c(C)noc1C.C(F)(F)F Cc1ccc(OC(F)(F)F)cc1C(N1CC(c2ccccc2)C(O)C1)=O c1(OC)ccc(NC(C2C(C)CCN2C(c2ccc(N)cn2)=O)=O)cc1C S(=O)(=O)(c1cccc(Br)c1NCc1ccc2c(c1)nc(C)n2O)NC c1(C(N2C(C)CCC2C(=O)NCc2ccc(F)cc2F)=O)cc2sccc2[nH]1 N1(C(CCC=C)=O)CCCC1C1CCCN1C(c1cncc(Cl)c1Cl)=O c1(OC)ccc(CC(N2CC(N3CCN(C(=O)C(O)C(C)C)CC3)C2)=O)cc1Cl C1(C(=O)NCC=CCNC(C2(F)CCCN(C)C2)=O)CCc2nccn2C1 C1(=CC(=O)NCC(C)NC(C2(O)CC(CF)C2)=O)CCN(C)C1 c1(CC)ccc(CC(=O)NC2CC(F)(CNC(=O)CC(C)SC)C2)c(F)c1 c1(CN(C(=O)Cn2nc(C(F)(F)F)cc2C(F)F)CC)nc2ccccc2n1C c1(C(N2C(CN(C(CN(C)C(N)=O)=O)C3CC3)CCC2)=O)cc(Cl)cc(Cl)c1N CC1CC(C(=O)NCC2CC2NC(c2cccnc2Cl)=O)CC(C)(C)C1 Cc1c(C(=O)NC(c2nc(C(N3CCCC3CC(C)(C)C)=O)co2)C)ccn1C Cc1ncccc1CNC(C1CCC(C2CC2)N1C(=O)CC(C)(C)N(C)C)=O c1(NC2(CN(C)C)CCC(F)(F)CC2)cc(=NCC#CCO)[nH]cn1 N1(C(Cn2ncc(CC)c2)=O)CCC(O)(CCNC(=O)CCC(=O)OC)CC1 C=C(C)CCCC(=O)NCC1(NC(=O)C=CC(=O)Nc2cnn(C)c2)CCCC1 c1(C(N2CC(CNC(C(CC)(C)O)=O)OCC2)=O)cc2ccccc2n1CC1CC1 C1(NC(CCC(=O)N(C(C)C)C)=O)CC2CCC1CN(C(=O)CO)C2 c1(C(=O)NC(C)C=CC(=O)N(C2CC2(C)C)C)ccn2ccccc12 C1(C(=O)NCC2CCO2)CC(O)CN1C(c1ccnc(Cl)n1)=O C1(NC(C2C(NC(Cc3ccc(C)nc3)=O)C2)=O)CCCOC12CCC2 c1(CC(=O)NCC(CNC(C(C=C)(C)C)=O)(C)O)c(C)[nH]c2cc(OC)ccc12 N1(C(C2N=C(C)SC2)=O)CC2(CCN(C(=O)CN(C)S(=O)(=O)N(C)C)C2)C1 C1(NC(c2ccccc2)=O)CN(C(c2csc(C(F)F)n2)=O)Cc2ccnn2C1 C1(CCNC(c2n(CC)ncc2)=O)CC(F)(F)CN1C(=O)CN(C)C(C)=O Cc1cc(CN2CCN(C(=O)NC3(C(F)(F)F)CCC3)C(C)C2)cc(C#N)c1 CCC1=C(C(=O)N2CCC3CCC(C2)N3C(c2ocnc2C2CC2)=O)SCCO1 c1(C(N(CCC)CCNC(=O)C(=O)NCC(F)F)=O)cc(S(N)(=O)=O)co1 c1(C(N2CCN(Cc3cccn4ccnc34)C3CC23)=O)cc(Cl)cc(Cl)c1O S(=O)(=O)(CC(=O)N1CCC(CNC(C2(C)COC(=O)C2)=O)CC1)NC c1(OC)ccc(NC(=O)C(N2CCOC3CC23)c2cocc2Br)c(C)c1 C1(CN(C(=O)COC2COC2)C)CCC(CNC(=O)CCc2ccoc2)CC1 CCC(C)CC(C(=O)O)NC1CCN(C(=O)CCCc2nc[nH]n2)CC1 CCC(C)C(C(=O)NC1(C)CS(=O)(=O)C1)NC(=O)C(C)CC(F)F C1(NC(c2nnnn2C2CCCCC2)C)CNC(=O)C(C)(C)C1 c1(C(N(CCCNC(C2(C)CCCC2O)=O)CC)=O)ccc(Cl)c(F)c1F C12(CNC(C3C(C)CCCN3)=O)CCCC1C2(F)F C1(NC(CC(COC)C)=O)COC2(C1)CN(C(c1cc(O)cc(Cl)c1Cl)=O)C2 C1(C(N2CCC(=C)CC2)=O)N(C(C2CC3(CC3)C2)=O)CCCC1(C)C C1(C#N)(NCc2c(N(C)C)cccc2)CCN(C(c2cc(C3CC3)n[nH]2)=O)C1 c1(C(=O)NCCC(C)CCNC(=O)Cn2cc(Cl)cn2)cc(F)c(F)cc1F C1(F)(C(=O)OCC)CCOCC1.C(CC(=O)NCC1(CC)CC1)N(C)C(=O)C1CC1 Cn1ncc2cccc(-n3cc(C4CCCN(CC5(C)CC6CC6C5O)C4)nn3)c12 C(=O)(C(F)(F)C(C)(C)O)NCC1CCCN(C(C(CC)Cc2ccccc2C)=O)C1 N1(C(c2c(F)ccc(C)c2)=O)CC2CC(NC(c3ncc(Cl)cn3)=O)CC2C1 N1(C2C(CC(=O)OC)CC2)CCC(C)(CNC(=O)C(C)NC(c2cccs2)=O)C1 N1(C(C2ON=C(CC)C2)=O)CCC2(CC2NC(=O)CC2COCCOC2)C1 Cc1c(OCCCN(c2nnnn2C)C)cccc1Cl.C1(C)CCSC1 N1(C(Cc2c(C)ccs2)=O)CCC(CNC(=O)CSCC2CCCO2)C12CC2 c1(C(=O)NC(CCOC)CNC(=O)Cc2ccsn2)cc(F)cc2cc[nH]c12 C1(C2CN(C(C3(F)CCCC3)=O)C2)(NC(C(C)NC(C2CCCC2)=O)=O)CC1 CC(CCNC(=O)CONC(=O)OC(C)(C)C)N(C(=O)CC1(C)CC1)C N1(Cc2c(C)ccc(C)c2O)CCC2(CCCC2C(=O)NC(C)(C)C)C1 C=CCC(CNC(=O)Cc1cn(C)nc1C)C(=O)NCCN1CCCC(O)C1 c1(C(N2CCOC(CNC(C34CCC(C3)C4)=O)C2)=O)ccc(CCF)cc1 n1(CC(=O)NC(CNC(CCN(C(C)=O)C)=O)(C)C(C)C)nc(O)ccc1=O C=CCC(CC)C(=O)NCC12CC(C1)C(NC(c1ccc(C(=O)OC)s1)=O)CO2 N(C(=NCCCc1ccccn1)N1CCC2(CCCC2)C1)CC(C)C#N C=CCC(CC)C(=O)N1CCN(C2CCCN(C(C3C4(CC4)C34CC4)=O)C2)CC1 c1(C(N(CC(C)NC(C(C2CC2)OC)=O)C)=O)cnc(C2CCC2)nc1O c1(CC(=O)NC(C)C(C)(C)NC(C2CCCC2OC)=O)cccc2c1CCC2 C1(C(=O)NCCOCCCN(C(CC(C)SC)=O)C)CC2(CCCCO2)C1 C(C=CC(=O)NCCC)(CC)=CC.C1(=O)CCO1 N1(C(=O)Cc2c(O)ncnc2O)CCC2(CCCN2C(=O)CCOC2CC2)CC1 C1(C(N2CC(NC(c3cncc(NC)c3)=O)(CO)C2)=O)CC(C)(C)CC(C)(C)C1 N1(C(C=Cc2n(C)ncc2)=O)CCC(NC(=O)Cn2nccn2)C(CO)C1 C(CS(=O)(=O)CC(=O)N1CCN(C(c2cncs2)=O)CC1C1CC1)OC C(=O)(C(C)(C)C1CCCCC1)NCCCOCC c1(C(N2C(C(=O)Nc3cnc(SC)nc3)CC3CC32)=O)cnc2c(c1)CNCC2 CCCCC(C)(C)NC(=O)C(C)N(C(=O)CC=CC(C)(C)C)C1CC1 C(C)(c1cnn(C)c1)=CC(=O)N(CCC(C)NC(C1(C=C)CC1)=O)C N1(c2c(C#N)cncc2)CC2(C1)C(NC(c1cccc(=O)o1)=O)CCS2(=O)=O C=CCC(C)N=c1nc2c(ncn2C(C)C)c(NCC(C)Cc2ccccc2)[nH]1 C#CCC(C(=O)OC)NC(c1cc(CNC(c2ccc(SC)o2)=O)nn1C)=O c1(OCCNC(C(=O)N(C)Cc2onc(CC)n2)=O)cccc(Cl)c1Cl C1(NC(=O)COCC2CC2)CCC2(CCCN(C(c3cnc[nH]3)=O)C2)C1 Cc1cc(C(=O)NCC23CC(NC(=O)CC4CCCCC4C)(CO2)C3)nc(C)c1 C1(C(N(CCNC(=O)C(C)(CO)NC(C)=O)CC)=O)CCS(=O)(=O)CC1 C(C)(CCCCCO)NC(C1C(CC)N(C(=O)CSCCC#N)CC1)=O Cc1ccc(C(=O)NC2(C)CC(NC(C3CCOC3C)=O)C2)c(N)n1 c1(CC)c(C(N2CC(NC(c3cn(CCO)nn3)=O)C(C)C2)=O)csc1C c1(C(N(CCNC(CC(C)CF)=O)CCOCCO)=O)cncc2nc(O)[nH]c12 C1(C(=O)NCCCN(C(C2(C)CCNC2=O)=O)CC)CC(S(C)(=O)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C)CC1CN(C(=O)C(F)C2CCC2)CCO1 N1(C(C(C)C2CCC2)=O)CCc2ccc(C(N3CCOC4CCCC34)=O)nc2C1 CC(C)(C)CCCC(=O)NCC1CC(C)(C)CN1C(c1ccc(S(C)(=O)=O)o1)=O N1(Cc2ccc(COC)[nH]2)CCCC(CNC(c2nc(C)sc2C)=O)C1 N1(C(c2cc(C)sn2)=O)CCC(C(CO)NC(c2oc(C(C)C)nc2C)=O)CC1 N(C1COCc2cccnc21)C1(c2n(C(C(C)C)C3CCC3)nnn2)CCOC1 CC(CCC(C)(C)C)C(=O)NC(CO)CCCCNC(c1cc(Cl)c(Cl)s1)=O N1(C(C(CCC)C#N)=O)CC(NC(c2cccc([N+](=O)[O-])c2)=O)CC(C)(C)C1 Cc1cn2c(n1)CC(C(N1C3CCC1CC(NC(=O)C(C)(C)CO)C3)=O)CC2 C1(CNC(C(C)=C(C)C)=O)CC(NC(c2cc(C(C)(C)C)no2)=O)CC1O c1(C(C)C)nc(NCCc2cccs2)cc(=NCC(F)(F)C(F)(F)Br)[nH]1 N1(C(c2ccn(CC)n2)C(=O)NCCCC)CCCCCC1c1cccc(F)c1 C(=O)(C(CCC)C(C)C)NC(CC#C)(C)C(=O)N1CCC(CC(C)(C)C)C1 C12(COC)CC(NC(=O)OC(C)(C)C)(CN1C(C1CC1c1cccc(C)c1)=O)C2 CCC(CC1CCCC1)C(=O)N1CC2CC2(NC(=O)CN2C(=O)CCC2=O)C1 C(=O)(C1=CCCSC1)NC1C2CN(C(C(CC#C)C)=O)C1C2 CON1CCC(CC(N2CCC(NC(c3csc(C)c3OC)=O)CC2)=O)CC1 c1(NC(C(c2ccc(Cl)cn2)N(C(CC)C)C)=O)ccc(F)cc1C c1(C(C(N2CCC(CC(=O)N(C3(C(N)=O)CC3)CC#C)C2)=O)=O)ccc(C)cc1 N1(C(Cc2snc(C)n2)=O)CC(C)(C)OCC1CNC(=O)C(C)c1ccsc1 N1(CCN(C(CC2CN(C(C)=O)C2)=O)C)CCN(C(C2CSCCS2)=O)CC1 N#Cc1sc(C(=O)NC2COCC2NC(C2CCCC3(CC3)C2)=O)cc1Br C(=O)(C1CCCc2cncn21)Nc1cccc(NC(C(COC)O)=O)c1 C1(C(=O)NCCC(C)N(C(C(=Cc2ccncc2)C)=O)C)CCCC2(CCC2)C1 CCCC(CC)CCC(=O)NC(C)C(C(=O)N1CCCCCC1)C(C)C C1(c2ccccc2)(NC(C(C)C2CCC2)=O)CC(NC(C2CCOC2)=O)C1 c1(CNC(C(CC)(C)C)C)cc(C(F)F)ccc1[N+](=O)[O-] c1(OCC(=O)NCCN(C(c2cccc(CC)n2)=O)CC)ccc(Cl)cc1F CCCC(C(=O)NC1CCN(C(c2nocc2CC)=O)CC1O)C(C)C C1(Cl)(C(N(CC(=O)NC2CCCC2)CCOC)=O)CC1C(C)=O CCCC(C(O)C(=O)N1CCCC(C)(C)C1C)NC(=O)C(F)OC(F)(F)F c1(C)ccccc1S(=O)(=O)NC(C1CCCCN(OC)C1)=O.C(C)(C)(C)S c1(OCC)cc(C)ccc1CNc1ccnc(N2CC(CC(=O)OC)C2)n1 N1(CC)CCC(n2ccnn2)C(O)C1.C(=O)(C(C)(C)CC#C)C1C(c2c[nH]nn2)C1 C1(F)(NC(n2ccnc2C)CC)COCCN(C(=O)OC(C)(C)C)C1 N1(C(c2cc(C)c(Br)o2)=O)CC(C)N(C(=O)C2=NOCC2)CC1C c1(C(N2C3(CNC(C(CC)(F)F)=O)CC(C2)C3)=O)cc2cc(Cl)ccn2n1 N1(C(C(C)N(C(C)=O)C)=O)C2CCC1C(C(=O)NC1CCCN(C)C1)C2 N1(C(c2c(C)occ2)=O)CCN(C(=O)CCC(C)(F)F)C(C2CCCC2)C1 C1(OC)C(F)CCC(C(=O)N(CCO)Cc2c[nH]nc2C)N1C(=O)OC(C)(C)C c1(C(=O)NC2CC(O)CN(C(=O)Cc3nc[nH]n3)C2)ncn2c(Br)cccc12 N1(C(C2(C)CSC2)=O)CC2(CC(C(=O)Nc3csnc3C3CC3)CO2)C1 N1(C(COC)=O)CCC(C2CN(C(=O)C(c3c(F)cccc3F)N(C)C)C2)CC1 c1(C(=O)NCC2C(NC(CN(C(C(C)C)=O)C)=O)C2)cnn(-c2ccccc2)n1 C1(NC(C2(CC#C)CC2)=O)CC(O)CN(C(c2ccc(-n3cccn3)cc2)=O)C1 c1(NC(C2(OC(C)=O)CC2)=O)ccc(S(=O)(=O)F)cc1 C#Cc1cc(C(=O)NC(C2(O)CCC2)C)ccc1Cl C1(NC(CSC)=O)CCCCN(C(=O)CNC(c2ccc(C)s2)=O)C1 CCCCC(CC)CC(=O)N1C2CCC1CN(C(c1cc[nH]n1)=O)CC2 C1(CC(=O)NC(C)(CNC(=O)CCOC2CCCC2)C2CCC2)CCOC1=O C1(NC(c2ncc(F)cn2)=O)CC2CCC1CN(C(c1ncc(F)cc1F)=O)C2 c1(CC)cc(C(N2CCC(C(C)NC(C3CCCCN3C)=O)CC2)=O)cc(Cl)c1 N1(C(c2c(CC=C)cccc2)=O)CC2C(NC(c3cncs3)=O)CS(=O)(=O)C2C1 C(=O)(C(C(=O)N1CCN(C(c2ccccc2Cl)=O)CC1C)C(C)(C)C)OCC C(C1CC(=O)N1)NC(c1nc(C)oc1C)=O.C(CCF)(C(=O)OC)COC N1(C(C(C)N(CC)CC)=O)CCN(C(=O)Cc2ccc(C#N)cc2)C2CCCC12 C1(C(N(CCCNC(C(Br)=C(C)C)=O)C)=O)OC2CCCCC2C1C C1(C2CC2)(C(N2C(C)CCC(NC(c3n[nH]cc3Br)=O)C2)=O)CCOCC1 c1(C2C(=O)O2)ccccc1.c1(CC)nc(-c2ccccc2)no1.C(C)(C)(C)O c1(C(=O)NCC2(F)CN(C(=O)COCC3CCOC3)C2)cc(C2CC2)ccc1Cl N(C1CN(C(c2snc(Cl)c2Cl)=O)Cc2ccccc21)C(=O)C1=CCCS1 CC1CCCC(C(N2CCCCC2CNC(=O)C(C2CCOCC2)C)=O)CC1 C1(C(=O)NC2CC(F)(CNC(C=C(C)CN3CCOCC3)=O)C2)CC(C)(C)CO1 c1(COC)ccc(C(N2CC(CO)(NC(=O)C(C)NC(N)=O)C2)=O)o1 C1(CC)C(C(=O)NCCC2CC2C(=O)OC)CCN1C(=O)Cn1nc(C)cc1C C1(NC(c2ccc(NC(C)(C)C)cc2)=O)CC(NC(C2COC2)=O)C12CCC2 N12CCCC(O)(C1)C2.C1(C(=O)NC(c2ncc(C)o2)C)CC(=O)NC(=O)C1 c1(CNC(C2CN(C(=O)OC(C)(C)C)CCO2)C)ccc([Si](C)(C)C)cc1 c1(CC(N2C3CC(CNC(C(CC#C)(C)C)=O)C(C3)C2)=O)cc2ccccc2o1 Cc1cc(N)ccc1C(N1CCC(C)(CCNC(c2cc(C)c(C)s2)=O)C1)=O c1(C(=O)NCCNC(=O)Cc2cc[nH]n2)ccc2c(c1)NC(=O)CS2 N1(C(C(C)(C)C2CCCC2)=O)CC(C2CC2C(=O)NC2CC3C=CC2C3)C1 C#CCC(C)(C(=O)N(C)Cc1cnn(C)c1)NC(=O)C(C)OC1CCCC1 Cc1cc(C(N2CCN(C(=O)C(O)CC(C)C)CC2c2cn[nH]c2)=O)[nH]c1C#N C(C)(CNC(c1coc(C(C)C)n1)=O)(CC(C)C)NC(C(CC)OC)=O Cc1cccc(CNC(c2conc2C(C)NC(=O)CCCF)=O)c1 C1(CNC(C(C)n2cncn2)=O)(CNC(C2CCOC2C)=O)CCCCC1 N1(C(=O)Nc2sc(NC(CCc3c(C)ccnc3)=O)c(C)n2)CC(C)OC(C)C1 c1(C(=O)NCC(C2(O)CN(C(C3CC3C(F)F)=O)C2)(C)C)c[nH]cc(Cl)c1=O c1(OC)cccc(C2CC2)c1.N1(CCOC)CCN(C(=O)CCSC)CC1 c1(C(=O)NCC(CC)NC(C2(Cl)CC2)=O)cnccc1C CC(C)CCS(=O)(=O)c1ccc(NC(=O)CC2COCCN2C(C)=O)cc1 Cc1cccc(Br)c1NC(=O)CC1CCCN1C(c1cc(F)n(C)n1)=O Cn1cc2c(C(=O)NC34CC3CN(C(c3cccc(C#N)c3)=O)C4)cccc2n1 N1(C(c2c(C)ccc(C)n2)=O)CC2CC1CN(C(=O)CSc1ccc(O)cc1)C2 c1(CCC(=O)N(CCC(=O)NCCC2CC2C)CC)nc(=N)[nH][nH]1 CCC(CC(=O)NCc1ccc(N2CCCCC2)cc1)C(C)C C#Cc1cccc(C(N2CCC(OC(C)C(N3CCC(=C)C3)=O)C2)=O)c1 N1(C(C(C)OCCC=C)=O)CCCCC1CN(C)C(c1ccc(CC#N)cc1)=O C(=O)(CC(F)(F)C(F)F)N1C2CC(NC(C3CC3C3CCCC3)=O)(C2)C1 c1(OC)ccc(C(C)C)c(C(=O)N(CCCN(C)C(C23CCCCC2C3)=O)C)c1 CC1=C(C(=O)NCC(CNC(C2(C)COC(=O)N2)=O)C(F)(F)F)CCS1(=O)=O CC1(C)CC(CNC(=O)CC2CCC(O)C2)N(C(=O)CCCNS(C)(=O)=O)C1 Cc1cc(C(N2CCCOC(CCNC(=O)CCC3CC3(Cl)Cl)C2)=O)cc(O)n1 C1C(C)(C)CS(=O)(=O)N1.C1(O)(COCC)CCCN(c2cc(C)nc(C)n2)C1 c1(-c2nc(CCNC(=O)C(c3cnc(C4CC4)[nH]3)C3CC3)on2)ccc(Cl)cc1 C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)CC2CCC2)CCC1CO CCCCS(=O)(=O)CC(=O)NC1CCN(C(C2CCOC2)=O)CCC1CO C12(C(N3CC(CNC(C(C)SC)=O)C(C(F)(F)F)C3)=O)CCC(C)(CC1)CO2 C1(NC(c2c(C)cn(C)n2)=O)CC2(CCN(C(=O)CCc3ccc(N)cc3)C2)C1 c1(CN(CC(C)(C)C)CCCC)c(Br)cccc1Br C(=O)(C(F)(F)C(O)CC)N1CC(OC)C(NC(=O)C(C)(O)CC(C)C)C1 N1(C(C(CC)C#N)=O)CCC(O)(C(C)NC(=O)C=Cc2cccc(CO)c2)CC1 N1(C(c2c(NC(C3C(C)CCC3)=O)cccn2)=O)CC(=O)NC(C)C1 N1(C(CC(=O)OCC)=O)CCC=C(C(=O)N2CC(C)CCC2CC)C1 CCCCC(CC)CC(=O)NC(CNC(c1ccc(F)cc1SC)=O)CCCC C1(C(=O)OC(c2nc(CC)on2)C)C2CC1(c1ccccc1)CO2 c1(C(C(=O)NC(CNC(c2c(CC)n[nH]c2)=O)C2CCC2)(F)F)cccc(C)c1 c1(C(N2CCC(CN(C(c3nc(CC)sc3)=O)C)CC2)=O)cc2c(ccn2C)[nH]1 Cc1cc(=O)n(C)nc1C(=O)NCC1CCCC1NC(c1cc(O)n(C)n1)=O c1(CC(=O)N(C)CCOCCN(C)C(C2CCSC2)=O)noc2ccccc12 N1(C(CCCCC)=O)CC2CC(NC(=O)C(C)OCc3ccccc3)C(C2)C1 c1(CNC(C2(OC)CC2)=O)cccc(NC(C2(O)COC2)=O)c1 C1(C(N2CC(OC)(CNC(c3ccnn3C)=O)C2)=O)CCc2n[nH]cc2C1 Cc1cccc(C(N2CCOCC2CC(=O)NC2CC(N(C)C3CC3)C2)=O)c1F S(=O)(=O)(c1cc(C)cnc1NCCCC1CCOC1)N1CCCC(C(C)=O)C1 N1(C(CCCNC(=O)OC)=O)C(C(=O)NCc2cccs2)CC2CC12 CC1(C)C(CNC(C2CC3COCC3C2)=O)CCN1C(c1cnc(N)c(N)c1)=O CCCCC(CC)C(=O)N1CCC(NC(c2ccc(C3(C)CC3)cc2)=O)C(O)C1 C(CCCCCC(=O)NC12CCCC1CCC2)n1cc(C2CCN(C)C2)nn1 CC1CN(C(=O)CCSc2ccccn2)CC(C)N(C(=O)CCN(C)C2CC2)C1 Cc1ccc(C(=O)NC(C)(C)CCNC(C2CN3CCC2CC3)=O)cc1O O=C(N=c1cc[nH]c(CCCO)c1)NS(=O)(=O)CC1CC2(CCOC2)CO1 C1(OC(c2cnc(C(C)CC)s2)=O)CCCN(C(=O)C(C(C)C)NC(=O)NCC)C1 c1(OC)cc(C(=O)NC2(C)CCC(NC(C3(C(C)C)CC3)=O)CC2)c(F)c(Cl)c1 CC1C(NC(c2ccc(F)s2)=O)CCCN1C(c1ccc(=O)n(C)n1)=O C1(CC)CC(C(=O)NCC(C2CCCN2C(C2CC2COC)=O)(C)C)CC(=O)N1 C(=O)(C1CCc2ccccc21)N1CCC(CNC(CN(C)C)=O)C12CCC2 N1(C(C(c2cccc(Cl)c2)OC)=O)CC2(C1)CN(C(=O)CCC1CCC1)CCO2 Cc1ccnc(N2CC(CC(C)NC(=O)CC(N3CCCCC3=O)C)C2)n1 c1(C(=O)NC2C(NC(CC(CCC)(C)C)=O)CC2)nc2cncnc2nc1O C(CCCCCC(=O)NC1(CNC(=O)CC(=O)OC(C)(C)C)CCCCC1C)SC N1(C(c2cc(C)nn2CCO)=O)CCC(NC(C2CC=CCO2)=O)C(CO)C1 Cc1nnc2n1CCC(C(N1C(C(=O)N(C)C)CC3CCCCC13)=O)C2 CCC(C)(COC)CNC(=O)CC(C)CNC(c1cc(C(N)=O)co1)=O C(=O)(C(C)C(C)(C)C)NCC(c1ccc(OC)cc1)NC(=O)Cc1nocc1C c1(C(N(C)CC2OCCN(C(COCCCCC)=O)C2)=O)ccnc(C)c1C C1(NC(c2c(CC)csc2)=O)CC2CCCC(C1)N2C(=O)C(C(C)C)N(C)C c1(OC)cccc(O)c1CN1CCC(O)C(C(=O)Nc2cccc(Br)c2O)C1 c1(CCNC(=O)C=Cc2ccoc2)ccc(CNC(C2CS(=O)(=O)C2)=O)cc1 c1(OCCC(=O)NCCNC(c2coc(Cl)n2)=O)cccnc1 Cc1cc(O)cc(C)c1C(N1CC(NC(=O)C(n2nccc2C)C)C1)=O C1(CC(=O)N(CC(C)CNC(=O)CCNC(C2CCCO2)=O)C)CCC(C)(C)O1 C1(NC(c2ncn(C)c2)=O)CCN(C(=O)C(C)(C)C2CC2)CCC1CO Cc1c(CN(C2CCN(C)CC2)C)ccc(O)c1O C(=O)(CC(O)CC(C)(C)C)N(C)CC1(NC(c2c(C)ccc(OC)c2)=O)CC1 c1(C(N(CC(C)CNC(=O)C(=O)NCC(F)(F)F)C)=O)ccc(C(F)(F)F)nn1 Cc1ccc(F)c(CNC(C23CC(C(=O)NCC=CC4CCC4)(C2)C3)=O)c1.C(C=C)N c1(OC)ccc2c(c1)CCC2N(C)C(=O)CC1CS(=O)(=O)CN1 C1(NC(CCCOCC)=O)CN(C(=O)Cc2cccc3c2OCO3)C2(CCC2)C1 c1(C(N(C)CC2CCN(C(C(COC)OC)=O)C2)=O)ccc(N)c2ccncc12 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC1C(C)CN(C(=O)CC2CCCO2)C1 CCCCCCCC1CCCC1N(CC(O)CCN)CC(F)F C(=O)(CC1=CSC2=NCCN12)NCCC(C)NC(=O)C(c1ccccc1)=O C(=O)(CN=c1[nH]cnc(Cl)c1N)N1CC(C)C(n2cc(C(O)C(C)(C)C)nn2)C1 c1(COC)ccc(C(=O)NC23CC2CN(C(c2csc(C(N)=O)n2)=O)C3)cc1F c1(C(N(C(c2ccccc2)CNCCO)C)=O)ncncc1-c1ccccc1F CC(C(=O)NC1C=CC(C(=O)N(C(C(N)=O)C2CC2)C)C1)C(F)(F)F c1(CC(=O)NC(CC=C)CNC(c2cc(Br)c[nH]2)=O)coc2ccccc12 c1(CN2CC(CC(=O)Nc3ccccc3CO)OCC2)ccc2ocnc2c1 c1(C(C2(CO)CC2(F)F)NC(=O)NCC(C2CCOCC2)C)cccc(Cl)c1 C1(C(=O)Nc2c(OC)ncc(C)c2)CN(C(=O)OC(C)(C)C)CCC1(C)C C1(NC(=O)CC2CCCO2)CCN(C2CCN(C(C3CCCC3O)=O)CC2)CC1 Cc1nc(CC2CC2)oc1C(=O)NC1CCCN(C(=O)CCOC2CCOC2)C1 Cc1cc(C(=O)N(C2CCCC2)CCNC(=O)CCC2CC3CCC2C3)n(C)n1 c1(SC)cncc(C(=O)NC2CCCC2C(=O)NCC2(N3CCOCC3)CC2)c1 c1(C(N2C(C(C)NC(C(COC)(F)F)=O)CCCC2)=O)cc(C(F)F)cc(F)c1 C1(NC(Cn2c(C)c(Cl)cn2)=O)CCN(C(=O)Cc2ccns2)C12CC2 C(=O)(C(C)(C)CCCO)NCC(CN(C(c1ccc(C)o1)=O)C)O c1(CS(=O)(=O)Nc2ccc(OCCOC)c(Br)c2)cccc2c1OC(C)(C)C2 c1(C(C)C)nc(N2CC3CCC2C(NC(c2ccsn2)=O)C3)cc(C#N)n1 N1(C(C=C(C)C(F)F)=O)CC2CC(CNC(c3ccc(Br)cc3C)=O)CC1C2 CC(C)C(CCN(C)C(c1ccc(-c2nnnn2C)cc1)=O)NC(=O)C(C)O c1(CC(=O)NCC2C(NC(C(CCSC)O)=O)CCC2)cnc2ccccc2c1 c1(NC(=O)NC2C(c3cccc(OC)c3)C2)nc2c(s1)CC(C)CC2 C(CO)(CCCCNC(=O)C(C)(C)c1cccs1)NC(Cn1ncn(C)c1=O)=O C#Cc1ccc(CCC(=O)NCC2CN(C)CCN2C(=O)CCSC)cc1 Cc1cc(C(=O)NC23CC(C(=O)NCc4ccoc4)(C2)C3)ccc1Br N1(C(c2ccc(C#C)o2)=O)CCC(C(=O)N(C(C)CSC)C)CC1(C)C C1(NC(C2CC(C)(F)C2)=O)CCN(C(C2CCCCC2O)=O)CC1F Cc1cccc2nc(O)c(C(N3CCN(C(=O)CC4CCCO4)C(C)C3)=O)cc12 CCC(CC(=O)NC1(C(=O)NCC(=O)N(CC)CC)CCC1)C1CC1 N1(C(=O)NCc2cc(OC)c(Br)cc2F)CC(C)Sc2ccccc21 N1(C(C(CC)NC(N)=O)=O)CCCC(O)(CNC(c2cc(C(C)C)[nH]n2)=O)CC1 c1(C(N(CC(C)CNC(c2c(Cl)cnn2C)=O)C)=O)cc2c(ccn2C)s1 c1(C(=O)NC2CN(C(c3c(C)coc3C3CC3)=O)C2)cc(Cl)cc(F)c1Br n1(C(C)C)ccc2c(N3CC4(CC(NS(=O)(=O)C(F)(F)F)C4)C3)ncnc12 c1(CNC(COCCC)=O)ccnc(NC(C2(COCCF)CC(F)(F)C2)=O)c1 c1(COC)nc2n(n1)CCCC2NC(=O)C(=O)NCC1CCC(C)C1 C(N=c1[nH]cnc(NC2CN(CC(c3ccccc3)C)C2)c1C)c1nnc(C)o1 CCCCC(CNC(=O)Cc1cccc(OC)n1)NC(=O)Cc1c(C)cnn1C CC1CN(C)CC1N=c1[nH]c(N(C)CCN(c2ccccc2)C)nc2ccsc12 c1(C(N2CCCC(C(=O)Nc3ncc(C#C)nc3)CC2)=O)ccc2ccsc2c1 C1(CC(=O)N(C)CCO)CC2(CC2)CN1C(C1C(C)(C)C1(F)F)=O c1(C(=O)NC2CCC(CNC(CN(CC(C)(C)C)C)=O)C2)nc[nH]c2nccc1-2 N1(C(c2c(CC)noc2C)=O)CC2CC1CC2N1CCC(C(N)=O)CC1 c1(C(N(CC(CNC(C(C)OCC)=O)(C)C)C)=O)cc2ccncc2cc1F N1(C(C(C(C)C)(C)O)=O)CCC(NC(c2cc(Cl)sc2Cl)=O)C2(CCC2)C1 CC(CC(F)(F)F)C(=O)NC1CCCC1NC(c1cnc2n1CCS2)=O c1(SCC)ccccc1C(=O)NC(C1CCN(C(=O)Cc2cnc(C)[nH]2)CC1)C C(Cc1cc[nH]n1)(C(=O)NCCc1ccccc1)NC(C1CN(C)C1)=O N1(C(C2C(C(C)NC(c3ccc(NC)cc3)=O)C2)=O)CCC(C)(F)CC1 Cc1csc2ncc(C(=O)NC3CCCC(NC(=O)CCCC(C)(F)F)C3)n12 CC1C(CO)CCCN1C(=O)CCCCN(C(=O)CNC(=O)CC#N)C C(C(C)(C)CC(=O)NC1CC(C(C)NC(C2CCN2C(C)(C)C)=O)C1)OC c1(CNC(C2CC(O)CN2C(c2ccccn2)=O)=O)cccc2c1CCC2 CN1N=C(C(=O)NC(C(=O)NC2CC3CC2C(O)C3O)C(C)(C)C)CCC1=O C=CCC(CNC(c1cnc(C)nc1)=O)C(=O)N1CCN(CC)CC1C N1(C(c2cc(CC)nn2C)=O)CCCOC(CNC(=O)CC2(C)CC2(Cl)Cl)C1 C(C(CNC(=O)CCc1cncnc1O)S(C)(=O)=O)NC(c1c(CC)[nH]cc1)=O N1(CCC2C(OCC)(OC)COCC2)CCC2C(OC)C(C)(C)C12 C#Cc1ccc(Br)c(C(=O)N(CCNC(=O)C(C2CCOCC2)C)C2CC2)c1 C1(NC(C(C(C)(F)F)(C)C)=O)CCC2(CC1)CN(C(=O)CCc1cnc[nH]1)C2 c1(CC)nn(C)c(CC)c1C(=O)OCCc1ccc(Cl)c(F)c1 CC(Cn1cccn1)C(=O)N1CC(c2ocnc2CNC(C2(CF)CCC2)=O)C1 c1(C(=O)NC(C2(CNC(C3CCN(C)C3)=O)CC2)C)ccn(CCF)n1 CC1OCCN(C(C2CCCCN(C(c3ccccc3O)=O)C2)=O)C1C O=C(C#CC1CC1)NCC1CCN1C(=O)CC1OCCCO1 c1(C(=O)NCCN(C(c2cncc(-n3ccnn3)c2)=O)CC)[nH]c(O)nc1C C(=O)(C#CC1(C)CC1)NC(C(C)NC(C1(OC)CCSC1)=O)CO c1(C(=O)NCCCN(C(C2(C)CC2)=O)C2CC2)cncc2cnccc12 C1(COC)CCC(C(=O)NC2(CO)CN(c3nc(C(=O)OC)ns3)C2)C1 N1(C(C2CN(CC)C(=O)C2)=O)CCOCC(F)(CNC(=O)CC2CCCC2)C1 C(=O)(C(C)CC(F)(F)F)NC1CCC(N(C(C2CCN(C(CC)=O)C2)=O)C)CC1 C(=O)(C1=NOC2(CCN(c3ncc(Br)cn3)C2)C1)Oc1c(C)ccc(C)c1 C1(C)(CNC(c2c(CC)cns2)=O)CN(C(c2cc3sccc3[nH]2)=O)CC1C C1(NC(C(C(C)NC(c2ccc(CO)nc2)=O)C)=O)CCC(C)(C)CC1 c1(C(N2CC(CNC(Cc3nc(C)oc3)=O)OCC2)=O)nn(C)c(C)c1Cl C=CCC(C)(O)C(=O)NC(=O)C(C)(C)C.C12CCCCN1C(=O)C(C)C2 n1(C(C(=O)NC2CCCN(C(C=CCOC)=O)CC2)C)nc([N+](=O)[O-])cc1C C1(N(C(C(CC)F)=O)C)CCN(C(=O)C(=O)NC2CCCCC2OC)CC1 C=CCCCC(C(=O)NCC1(C)CSC(C)=N1)NC(c1ccc(NC)nc1)=O C(=O)(C1=CC2(CCOC2)C1)NCC1CN(C(C(C)(O)C2CCOCC2)=O)C1 c1(C(=O)NCCCN(C(C(CCSC)OC)=O)C(C)C)cnc([N+](=O)[O-])n1C C1(CNC(CC(=O)NCC)=O)CC2CCC1N(C(=O)C(O)CC1CCCCC1)C2 C1(NC(CCCC(=C)C)=O)CC2CCC1CC2NC(C1CC(OC)C12CCC2)=O N1(C(c2c([N+](=O)[O-])ccc(C)c2)=O)CCC2(CCCN2C(=O)CC2C=CCC2)C1 c1(C(=O)NCC(CNC(c2c(OCC)ccs2)=O)CO)sc(C)cc1Cl CCCC(CC)C(=O)NCC1CN(C(=O)CCCF)C1 C1(C(N(CCC(=O)NC2CC3CC3C2)CC#C)=O)CC12CCOCC2 N1(C(c2c(C)ccn2C)=O)CCCC2(CCN(C(=O)C(CO)C(F)(F)F)C2)C1 Cc1c(C(N2CC(N(C(=O)CC34CCC(CC3)C4)C)C2)=O)sc2ccsc12 N1(C(C(C)N2CC(NC(=O)OC(C)(C)C)C2)=O)CCc2c(O)n[nH]c2C1 C12(CCN(C(=O)CCCOC(C)C)CC1)C(=O)NC2.c1(CC)n[nH]c(C)c1C C1(CNC(Cc2cn(C)nn2)=O)CCN(C(C2CCCC23CCC3)=O)C1(C)C c1(C(=O)NC2(CC)CCN(C(=O)NCCCl)C2)ccc2cc(F)c(F)cc2n1 C1(NC(C2CCN(C(C(C)n3ccnn3)=O)C2)=O)CCN(S(C)(=O)=O)CC1 c1(OCC)ccc(C(=O)N(CCNC(C2CC(C)CO2)=O)C(C)C)cc1C c1(C(N(CC(C)(C)CNC(C2(n3cccn3)CCC2)=O)C)=O)cnc(N)cn1 n1(CC)ccc(CC(=O)N(C2CCCCC2)CCNC(C2COCCO2)=O)n1 C1(C(=O)NC2C(C)N(C(c3cccc(Cl)n3)=O)CCC2)CCC2(CCC2)CO1 c1(C(N(CCCNC(=O)Cc2ccon2)CCO)=O)cccc2c1CCO2 C=CC(O)(C(=O)N(C)CCNC(C12COCC1C2)=O)C(F)(F)F C1(NC(c2c(CC)cns2)=O)CCN(C(=O)CCc2cncs2)CC1F NS(=O)(=O)c1cc(C(=O)NC2CCC(NCC3CCC3)C2)ccc1Cl c1(CC(=O)NCC(C(C)C)NC(C2(C#N)CC2)=O)csc2nccn12 C(=O)(CCCC(=O)N1CC2CC1C2C(=O)Nc1cc(Cl)ccc1F)OC C1(F)(CN(C)C(=O)NC2CCCS2)CCCN(C(=O)C2=NOC(C(C)(C)C)C2)C1 CCC1=NOC(CC(=O)NC2CC(CO)(NC(C3CC(O)CN3C(C)=O)=O)C2)C1 S(=O)(=O)(c1cccc2c1OC(C)(C)C2)N1C(C)Cc2c(Br)cccc2C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC1CC2N(C(CCC#C)=O)C(CC2)C1 C=C(C)CC(C(=O)OC)NC(=O)CCCN(C)C(c1c[nH]cc1C)=O N(C(=NCc1ccccn1)NC1CCCC1(C)C)C1CC(C(=O)OCC)C1 c1(N(CCCN2CCCC2)C)nc(NCC2CCSC2(C)C)c2c(ncn2C)n1 C1(C(N)=O)(NC(=O)CC2NC(=O)CS2)CCCC1.C1(SCO)CCC1 c1(OC)ccc(C)cc1C(=O)NCC1CN(C(=O)CSc2ccncc2)C1 c12ccc(F)c(c1)COC2=O.n1(CCC)cc(C2CCCCC2)c(C2CC2)n1 N1(C(C2N(C(C)=O)CCC2)=O)CCOCC1CNC(=O)CSc1n[nH]c(O)n1 C#CCC(C(=O)NCC=C)NC(=O)CCNC(C1CCSCC1)=O c1(OC)cc(C2CCN2C(=O)N(C(C)C(C)C2CC2)C)ccc1C(F)F Cc1nnc(O)c(C(N2CCCC(O)(CNC(c3cnc(S)[nH]3)=O)CC2)=O)c1C C1(F)(CNC(CN2CCC(OC)C2)=O)CCC(CNC(=O)CNc2nccs2)C1 N1(C(c2cncc(COC)c2)=O)CCC2CN(C(C3(C(F)F)CC3)=O)CCC12 C1(CNC(c2cnc(SC)[nH]2)=O)CCCC(CNC(=O)Cc2ccc(F)nc2)C1 Cc1cccc(C(=O)C(=O)NC23CC2CN(C(=O)Cc2c(C)n[nH]c2C)C3)c1 C1(C(=O)NCC(C2CCCCC2)NC(c2ncn(C(C)C)n2)=O)CC12CC(O)C2 N1(CC(=O)NCCCn2cc(Cn3ccnc3)nn2)CCCCCS1(=O)=O C(=O)(C(C)(C)CN(C)C(c1ccnc(C(N)=O)c1)=O)NC(C1CCOC1)C#C CN(CCCC(=O)NC1CC2(CCN(C(c3sncc3Cl)=O)C2)C1)N=O c1(C(CNC(=O)Cc2nc(-c3ccccc3)n[nH]2)=O)ccc([N+](=O)[O-])cc1 c1(C(N2CC3CC3(CNC(C3(O)CCOC3)=O)C2)=O)cccnc1SC(F)(F)F C1(C(=O)NCC(C)CN(C)C(c2cnccc2Cl)=O)CCCc2ccccc2C1 CCCC(CC)C(=O)N1CCN(C(c2cc(C)[nH]n2)=O)C(CC(C)(C)C)C1 C(=O)(C(C)(F)C(=O)NC(CNC(=O)CCn1ccnn1)CC(F)(F)F)OCC c1(C(N2CC(N(C)C(c3sccc3CO)=O)C2)=O)cc(S(N)(=O)=O)ccc1F N1(C(C(c2cn(C)nc2)NC(C2CCCC(C)(C)C2)=O)=O)CCC(=C(F)F)CC1 N1(C(C2CCC(C)(C)O2)=O)CCC2C(C1)NC(=O)CN2C(=O)CCN1CCCC1 N1(C(c2c(C)cc(C)oc2=O)=O)CCCC(C2CCCN(C(C3(Br)CC3)=O)C2)C1 C1(N(C(c2cnns2)=O)CC)CCN(C(=O)CC2C=NN(C)C2=O)CC1 c1(CCNC(=NC)NC2CCN(C)CC2)ccc(C)nc1Br c1(OCC)c(C(N2CCOC(CNC(C3(CC)CC=CC3)=O)C2)=O)cccc1C c1(C(=O)NCC2(CNC(CC3CC(C)C3)=O)CCC2)ccc2cc[nH]c2c1 C(=O)(CCC(=O)N1CCCC1CN(C(C1CC(OC2CCC2)C1)=O)C1CC1)NC Cc1ccc2c(CN(CCN=c3cccn[nH]3)CCO)c[nH]c2c1 C1(NC(C(COC)COC)=O)CC2CC1N(C(=O)CCC1CCCO1)C2 c1(C(C(=O)NC2CC(NC(C3CCNC(=O)C3)=O)C2)(F)F)cccc(Cl)c1F c1(NC(CC2(NC(CC3C(CC)C3)=O)CCC2)=O)cnn2cccnc12 CCN=c1[nH]c(C)c(C(=O)NC(CNC(C2CCOC2C2CC2)=O)C(C)(C)C)s1 N1(C(C2(CC(C)C)CC2)=O)CC2(C(=O)NC(C)(C)C(C)(C)O)CCC1CC2 c1(C(N2CCC3(C(=O)Nc4cccc(N)n4)C(C2)C3)=O)cc2ccccn2c1 C(=O)(C(C(C)O)NC(C1CCC(=O)O1)=O)NCCOCC(=C)C Cc1nc(C)c(CC(=O)NC2CCC2CNC(c2cnc(O)s2)=O)s1 CC1(CC(N2CCC(CNC(c3ccn(C(F)F)n3)=O)C2)=O)OCCO1 Cc1cccc(C(=O)NC2(CO)CCSC2)c1Cl c1(C(N2CCC(O)(C(F)(F)CO)C2)=O)ccccc1Cn1cccn1 C(=O)(C(C)C(F)(F)F)NCC1(CNC(c2nccc(CC)c2)=O)CC1(F)F c1(C(=O)NCC2CC(NC(c3cc(Cl)no3)=O)C(O)C2)n[nH]c2c1CCCC2 Cc1ncnc(O)c1C(N1CCC(C)(CC(=O)NCC2(CO)CCCO2)C1)=O N1(C(c2cn(C(COC)C)nc2C)=O)CCN(C(=O)C(F)CCC)CC1CCO C(C(C)(C(C)C)NC(c1ccc(C)cn1)=O)NC(C1CC(C(=O)OC)C1)=O C(CC(=O)N1CC2CN(C)CC2C1)(CC(C)C)NC(C(C)NC(CC)=O)=O CC(C)CC(F)(F)C(=O)NCCC(C(C)C)NC(C1(C(F)(F)F)CCCC1)=O c1(OC)ccc(CCC(=O)N2CC(N(C)C(C3CC34CCC4)=O)C2)c(F)c1 C1(NC(C=Cc2ccc(C)s2)=O)CN(C(c2ccc(C)c(C)c2)=O)CC1C#N N1(C(c2nc(CNC(C(C)n3cncn3)=O)oc2)=O)CCC(C)(CO)CC1 C1(Cl)(C(=O)NCCCC(=O)N2CC(CN=[N+]=[N-])C2)CCCCC1 c1(C(=O)NC(C)CNC(=O)Cc2cscn2)cc(N)c(F)cn1 Cc1ccncc1C=CC(=O)NCC1CC1CNC(c1ccc(C(C)O)cc1)=O c1(C(=O)NC2C(NC(C(CCC)(C)C)=O)COC2)nn(C)cc1S(N)(=O)=O C1(NC(C(c2cccc(C)c2)C)=O)CCCCCN(C(C2(C3CC3)CCC2)=O)C1 C1(C(=O)OC(C)(C)C)CCCCN1C(=O)NC(c1cccn1CC1(O)CC1)=O.CN c1(C(C(=O)NC2CC2)N(C(C#C)C2CCC2)C)ccc(OC)o1.C(COC)C(C)C C1(CCC)CN(C(c2ccc(CC)nc2)=O)CCO1.C1(c2ccco2)C(=O)N1 C1(C(C)NC(C=CC=CCC)=O)CCCN1C(=O)CCn1cncn1 n1(C2C(NC(c3csc(C4CC4)c3)=O)CC2)cc(C2CCCO2)nn1 Cc1ccc(NC2CN(CCCCNC(=O)C3CC3)CC2C)cc1 CC1(C)CC(CNC(=O)CC23CCCC2C3)CN1C(c1cc(F)cnc1O)=O c1(C(=O)NC2C(CNC(C(C)(C)c3cscn3)=O)C2)cc(F)cc(F)c1 N1(C(Cn2ccc(C)n2)=O)CC2(CC(NCC(=O)NS(C)(=O)=O)C2)C1 N1(C(C2(C)CC2(Cl)Cl)=O)CC2CCC(C1)C2CNC(=O)CNC(N1CCCC1)=O C(=O)(C(C)CC(N)=O)NCCCCC1CN(C(CCC(C)OCC)=O)C1 C(CC(CC)C(=O)NCCN(C(C1CCCN(C(=O)C(C)(C)C)C1)=O)CC)=CC c1(C(=O)NCC2N(C(CS(CC)=O)=O)CC=C2)cc(Br)ccc1-n1cnnn1 c1(COC)nc(C)cc(=NCC2C3CN(C(c4ccc(CCO)cc4)=O)CC23)[nH]1 CC(C)CC(CC(=O)N1CC(O)CC1(C)C(N)=O)NC(c1cncc(O)c1)=O c1(OCCOC)nc(C)ncc1COC(C1CC12CC(N)C2)=O C(=O)(CCC(F)(F)F)NC1C2CN(C(C(CCSC)OC)=O)CC21 CC1c2ccccc2OCCN1C(=O)NC1(C(=O)NCCSCCN)CCCCC1 c1(N(C(=O)CC#N)C2(C3N(C(c4c(OC)scc4)=O)CCC3)CC2)c(C)coc1C C1(O)(CC(=O)NCCN(C(C2C(C)CC2)=O)CC)CCOC1 c1(NC(C2CC(C)N2C(c2ncoc2C2CC2)=O)=O)ccc(F)cc1 c1(C(N2CCOCC(NC(CC=C=C)=O)C2)=O)cnc(O)n(C)c1=O N1(C(CC2CCN(C)C2)=O)CCCCCC(NC(C2CC(=C(F)F)C2)=O)C1 C1(C(N(CCN(CC)C(C(C2CCCN2C(=O)OC)=O)=O)CC)=O)C2CC(=O)CC12 c1(C(N2CCN(C(C(C)OC)=O)CC2CF)=O)ccc2sc3ccccc3c2c1 c1(C(=O)NC(CN(C(=O)CC2(c3ccccc3)CC2)CC)C)cnc2nccn2c1 c1(OC)ccc(-c2nc(C)c(C(=O)NC3CC3C(=O)NC3(CC)CCC3)s2)cc1 N1(C(C2(NC(=O)C(C)NC=O)C(C)CCC2)=O)CC(N(C)C)C(C)(C)C1 c1(C(C(=O)OCc2scc(C(=O)OC)n2)OCC2CCCO2)ccncc1 C#Cc1cccc(C(=O)Nc2cccc(N(C(c3ncnn3C(C)C)=O)CC)c2)c1 c1(C(=O)NCCCC(C)NC(CC2(OC)CCCCC2)=O)nccc(OC)c1F C(=O)(CC(CNC(C1C2CCCC12)=O)C1CCC1)NC(C)(C)C C(CC(C(=O)N1CCC(N(C)C)C1)NC(=O)CC1CC2CCC1O2)N(C)C N1(C(Cc2c(C)occ2)=O)CCC(O)(CN(C(=O)C(C(C)C)n2cccc2)C)C1 N1(C(c2nc(Br)co2)C(=O)NCC2CCCO2)CCc2c(Br)ccc(F)c2C1 CN1C(=O)CCC1(C)CNC(=O)CCC1(NC(C23CSCC2C3)=O)CCCC1 Cc1nnc(O)c(C(=O)NC2CN(C(c3c(C)nc(C)nc3C)=O)C2)c1C C1(CNC(c2c(F)cccc2F)=O)CC2CC(C1)N(C(c1cc(O)ncn1)=O)C2 C1(O)(C(C)NC(c2ccccn2)=O)CCN(C(c2cc[nH]c(=N)c2Cl)=O)CC1 C1(NC(c2csc(C)c2Br)=O)CCN(C(=O)Cc2nncn2C)CC1O C1(NC(=O)CC)(CC)CCCN(C(c2cc(NC(C(CC)CC)=O)no2)=O)C1 C1(C(=O)NCCC(C)O)CC(N=[N+]=[N-])CN1C(=O)C=CCO C=C(C)CC(C(=O)N1CC(F)CC1C(=O)NC1CC1c1ccnc(O)c1)OC N#Cc1cc(C(=O)NC(CNC(=O)C(F)(F)C(O)C2CC2)C2CC2)cc(O)c1 c1(NCCNC(N(CC)Cc2ccc(O)cc2)=O)c(F)cc(Br)cc1F C(=O)(C(C)(C)C(C)(F)F)N(CC(O)CNC(C12CCCN1CCC2)=O)C c1(C(=O)NCC23C(CN(C(C(C)O)=O)C2)C3)cc(O)cc(F)c1F C(=O)(C(CNC(=O)Cn1c(O)nnc1O)C(C)(C)C)NC(CCC)C(C)(C)C C1(C(=O)NCC(CNC(C(c2cccc(C)n2)C)=O)(C)C)CCC(F)(F)C1O c1(N2C(CNC(C(CC)CC(C)C)=O)CN(C)CC2)ncnc2sc(C)nc12 Cc1noc2ncc(C(=O)NN3CC(CN)C3)cc12.c1(CC)cc(F)ncn1 c1(C(=O)OC(C(=O)OC)c2ccns2)cccc(NC(N)=O)c1 C12(CNC(N(C(CCC)(C)C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1C2 C(=O)(CC1OCCc2ccsc21)N1C2CN(Cc3cc(C)no3)C(CC2)C1 c1(C(=O)NC2CC(CCNC(c3cc(OCC)n[nH]3)=O)C2)cc(=O)c(CC)c[nH]1 Cc1[nH]c(=NCC(O)CNC(c2scnc2C(C)(C)C)=O)ccc1C#N c1(C(=O)NC(CC(C)C)CNC(C2C3COCC23)=O)ccc2nccn2n1 c1(SCC2C(C)CN(C(C3(S(C)=O)CCNCC3)=O)CC2)cccc2cc[nH]c12 C#Cc1cccc(C(=O)OC)n1.C12CCN(C1)C(=O)NC2 c1(C(=O)NC2C(C)CN(C(=O)Cc3nocc3Br)C2)cc([N+](=O)[O-])cnc1O Cc1cc(N(C)Cc2ncn(C)n2)nc(=NCc2ccc(Cl)c(F)c2F)[nH]1 CS(C)(=O)=Nc1ccc(C(N2CCN(C3CCCC4(CCC4)C3)CC2)=O)s1 c1(C(C(N2C(CN(C(C3C(C)(CC)C3)=O)C)COCC2)=O)C)cccc(C#N)c1 CC1CN(C(C2(C)C=CCN2C(C2CC3(C2)CC32CC2)=O)=O)CC(C)N1C C1(C(=O)NCC(N(OCC)C)=O)CN(C(c2cnc(CC)o2)=O)CC12CC2 C1(C(N2CCC(F)(CO)C2)=O)(CNC(C2C=CCCCC2)=O)CCCCC1 N1(C(CC2(CNC(c3c(CC)n[nH]c3)=O)CC2)=O)CCOCC1CCF Cn1cc(C(N)=O)cc1C(N1CC(O)(CNC(=O)C(F)F)C1)=O Cn1cc(C(=O)O)c(C2CCCN(CC3(C)COC(=O)N3)C2)n1 C1(C(=O)NC2C(NC(C3(CC)CC3)=O)CCC2)CCCC(C)(C)O1 CC1(C)CCC(CC(=O)O)(NCCS(=O)(=O)NC(=O)OC(C)(C)C)CC1 C1(NC(C2(CCC=C)CC2)=O)CN(C(C2OCCOC2C)=O)C2(CCC2)C1 C(=O)(CC(O)CC(C)C)NCC(CN(C(c1ccc(C(F)F)o1)=O)CC)(C)C c1(C(=O)NC2C(NC(CSc3c(C)cccc3)=O)CC2)c[nH]cc(F)c1=O Cc1cncc(C(=O)NCC2CCN2C(=O)C(c2ccc(F)cc2)C)n1 Cc1nsc(C)c1CC(N1CCC(NC(c2cc(C)n(C)c2)=O)C1)=O c1(C(CC(=O)N2CC(CC(=O)OCC)C2)NC2(C)CCCOC2)ccccc1F N1(C(c2cncc(C)n2)=O)CC(C(N2CCCC(C)CC2)=O)CC1(C)C c1(C(N2CC(C)(NC(C3(C(=O)OC)CC3)=O)C2)=O)cnc2ncccc2c1 N1(C(c2scc(C)c2)=O)CCC(C(=O)NCC2(CN(C)C)CC2)CC1(C)C C1(CC#C)(C(=O)NCC(C)NC(c2ccncn2)=O)CCCOC1 C1(C(=O)C(OC)=O)CCCC1.c1(C(=O)OC)c[nH]nc1CCNC1(C2CCCC2)CC1 N1(C(c2c(C)n(C)nc2)=O)CC2(CCC2)CC1C(=O)NCC1(CO)CC2(CC2)C1 C(=O)(C(C1CC1)NC(C1CC(SC)C1)=O)NCCOC C1(C(=O)Nc2cncnc2O)CCN(C(=O)CC2CSCCO2)CC1O C1(C(=O)NCC(CNC(c2cc(CC)no2)=O)OC)CCC(=O)N(C2CC2)C1 C1(NC(C(c2cccc(F)c2)C)=O)CC2CN(C(C3COC4COCC34)=O)CC12 C1(CCNC(C2C(=C)C2)=O)CN(C(c2cc(C)nnc2O)=O)CC(C)O1 c1(C(=O)NC(CCCOC)C(=O)N(C)Cc2noc(C)n2)c[nH]c2nccc-2c1 C(=O)(C(C)(C)c1cc[nH]n1)N(CC1(C(C)NC(C2COC2)=O)CC1)C1CC1 c1(C(N2C(C)CCC(NC(CCOCC#C)=O)C2)=O)cc2cc(F)ccc2cn1 C(=O)(C1=CCC(F)(F)CC1)N1CCCCC(NC(Cc2c(C)ncs2)=O)C1 Cn1cnc2c1CN(C(C1CN(C(c3csc(Cl)c3)=O)CCO1)=O)CC2 N1(C(C(N=S(C)(C)=O)=O)=O)CCC2(CC1)CN(C(=O)CCc1cccnc1F)C2 O=C(C1=CC2(CCOC2)C1)NCC1C2CN(C(c3nc4sccn4c3Cl)=O)CC12 c1(C(N(C)CC2(O)CCN(C(C3CN(C)C3)=O)C2)=O)cccc(Cl)c1F Cc1nc(N2CCC(C)C(NC(=O)C=Cc3cccc(Cl)c3)C2C)cc(C#N)n1 c1(OC)ccc(F)c(C(N2C3CC2CN(C(c2sc(Br)nc2C)=O)C3)=O)c1 c1(C(N(C2CCN(C(CC(CC)C)=O)C2)CC)=O)nc(O)nc(O)c1F CCCN(NC(=O)CCCCc1cnc[nH]1)C(N)=O.C12CC(C1)N(CC)C(=O)C2 C1(C(=O)OCC)(CNC(C2(CNC(C(Br)=CCC)=O)CC2)=O)CCOCC1 N1(C(CC2CN(C)CC2O)=O)CCN(C(=O)CCN2CCCC2)C2CCC12 CON(CCC(=O)NCC(C)(C)OCCO)C(=O)c1nc(=N)cc[nH]1 CC(C)C(C)CC(=O)N1CC2CC1C2C(=O)N(C)CC1CCOC1C N1(C(C(C=C=C)C)=O)CCN(C(c2c(CC)ncnc2CC)=O)CC1CC CC1(C(=O)Nc2cccc(-n3cc(C4C5CC6C(C5)C46)nn3)c2)CC(C#N)C1 C1(C(=O)NCCCNC(CC)=O)CN(C(=O)C(C)N2CCC2)C2(CCCC2)C1 C1(COC)(CNC(=O)CCCNC(N)=O)CCCN1C(=O)C(C)N(C)C CCC(CC(=O)NC(C)CCNC(=O)C(C)(C)OCCOC)CC(F)(F)F Cc1c(NC(c2cccc(CNC(=O)CSCCC(F)(F)F)n2)=O)nnn1C C1(C)(OC)CCN(C(C2C(C)CN2C(=O)CC2(O)CCCC2)=O)C1 Cc1nn(C)cc1CN(C(=O)CC1CN(C(C2(C)CC(C)C2)=O)CCO1)C N1(C(C(CC(C)C)O)=O)CCC(C)(C)C(CNC(=O)C(C)OCC(F)(F)F)C1 CN1CC(C(=O)NCC2COC(CNC(=O)CCCC3CCCO3)C2)NC1=O n1(CCC2CN(C(=O)Cn3ncnn3)C2)cc(-c2cncnc2)nn1 C1(C(=O)NC(c2ccccn2)CC)CCCN1C(=O)CSCC(N1CCCC1)=O C1(CNC(c2cnc(CCC)s2)=O)CN(C(=O)C(C)(C)CC)CCC12CCOC2 N1(c2cc(C)ncc2C#N)CCC2(CNC(=O)CCCC(F)(F)F)CCCCC12 c1(OC)c[nH]nc1C(=O)N(C)CC1(NC(=O)CC2CCOC2=O)CC1 CC1CCN1CCN(C1CN(C(=O)CC=CC(C)(C)C)C1)C N1(C(C(C)NC(C)=O)=O)CC(F)(N)C1.C(=O)(C(C)OC1CCOC1)SCC.C1CO1 C1(OC)CC(CC(=O)N(CCC(C)NC(=O)C2=CCCC2)C)C1(C)C C1(C(N(C(CCC)C)C)=O)CCN(C(=O)C(c2ccccc2)C)C(C)(C)C1 CC1CCOCC1C(N1CC(O)(CNC(c2nccnc2N)=O)C1)=O N1(C(C2C(C(C)(F)F)C2)=O)CCN(C(=O)CC2(C(F)(F)F)CCC2)CC1CO c1(CC(=O)NC2C(C(=O)OC)COC2)cc(=O)n(-c2ccc(Cl)cc2)[nH]1 N1(C(CC2C(OC)COCC2)=O)C2CCC1CC(N(C)C(C1(C(F)F)CC1)=O)C2 N1(C(C2(C)CCC2)=O)CCOC(Cn2cc(-c3ccc(Cl)cc3)nn2)C1 c1(OCc2ccc(C(C)(C)O)cc2)cccc(CSC)c1.CCC1CN1 CC1CN(C)CCC1NC(C1CCC1c1ccc(F)cc1)=O N1(C(c2c(OC)nccc2)=O)CCN(C(C2(F)CC=CC2)=O)CC12CCC2 c1(C(=O)NCC#CCNC(C#CC(C)C)=O)ncc(F)cc1F C1(C(=O)NC2C(C)OCCC2)CC2(CCN(C(C3(C#N)CCC3)=O)C2)C1 c1(C(=O)O)cc(S(=O)(=O)NC(c2nc(C3CCCOC3)cs2)=O)ccc1F c1(C(N2CC(NC(CCSCCC)=O)C(SC)C2)=O)sc2nccc(C)c2c1C CC1CN(C(C2COCCO2)=O)CC1CCNC(c1cc(C2CC2)[nH]n1)=O C(CC(O)C(=O)NCCOCCCN(C)C(C1CCN1C)=O)SC C1(c2ccccc2)(NC(F)F)CCN(C(=O)NCC(C)C)C1 c1(CNC(C2N(C(c3nc(CC)oc3)=O)C(C)C2)=O)ccc(C)c(C)c1 N1(C(CCC(C)C)=O)CCN(C(c2cnc(O)c(F)c2)=O)C2CCCC2(C)C1 C1(NC(c2ccc(NC(=O)CO)cc2)=O)COC2(C1)CN(C(CCCCS)=O)C2 Cc1nc2ccc(O)cc2cc1C(=O)NC1CCN(C(C2CCC(=O)NC2)=O)C1 C1(OC)CC(NC(=O)CCN2CCN(C)CC2)CN(C(=O)CCCC2CCC2)C1 C1(CN(C(=O)COC2CCC2)C)CCCN(C(c2cnc(C(C)(F)F)s2)=O)C1 N1(CC)CCCC(C(=O)N(CC(=O)NCCC2CC(O)C2)CC(C)C)C1 N1(C(c2c(C(C)NC(C3(CCOC)CC3)=O)noc2)=O)CCCC2OCCC2C1 c1(C(=O)NCC2CCC(C(=O)NCC3ON=C(C)C3)C2)cc(C#N)ccc1C Cc1nc(=N)[nH]c(C)c1C(N1CCN(C(=O)Cn2cc(Cl)cn2)C(CCO)C1)=O c1(CNCC(C2(OCC)CCCC2)(F)F)cnc(C)n1C(F)(F)F n1(CC(N2CCC(CN(C)C(C3C(F)(F)C34CC4)=O)CC2)=O)ccc(O)nc1=O O=C(C#CC1CCOC1)NCc1nocc1C(=O)NC(C(F)(F)F)C1CC1 N1(C(CCC)=O)CCCCC1C(=O)N(CC(C)NC(C)=O)C C(=O)(C(=O)N=S(C)(C)=O)NCC1(C)CCC(NC(C(CC=CC)C)=O)CC1 C1(CC=C)(C(=O)NC(C)CC(C)NC(c2cc(C(C)(C)C)no2)=O)CCOCC1 N1(C(C2C(OCC)CC2)=O)CCC(C=CC(=O)NCC(C)O)CC1 C=CCC(Cc1ccccc1)NC(=O)NCC(C)(O)CCO c1(C(=O)NCc2ccc(CCNC(C(CSC)O)=O)cc2)ccc(O)cc1C C(C(C)(C)C(=O)NCC1CC(F)(F)CO1)N(C(C1CC(C(C)C)C1)=O)C C1(CNC(=O)CC2(O)CCC2)CC2(CCC2)CN1C(C1CC1C(F)(F)F)=O C(=O)(C(c1ccoc1)NC(=O)C(C)SC)NCCN(CCC)C(C)C C(C(C)C(F)C(=O)NCC1CC=CCC1)NC(c1c(C)scc1)=O N1(Cc2c(C)ncs2)CCC2(CC1)CC2NC(c1cc(O)cc(F)c1)=O CC1CC(NC(c2ccc(C3CC3)s2)=O)CCN1C(=O)CNC(c1cccnc1)=O C(=O)(C(O)CC(F)(F)F)NCc1c(C(N(CC(C)(C)C)CC)=O)scc1 C1(CNC(C2CC2F)=O)CN(C(=O)CC2CCS(=O)(=O)C2)CCC1(F)F Cc1nc(NCCSC(C)(C)C)cc(Nc2ccc(C(C)(C)C)cn2)n1 Cc1c(C#N)c(N2CCC(N3CC(C)OC(C)C3)CC2)nc2ccccc12 C1(NC(C(F)=C(C)C)=O)CN(C(=O)Cc2c(Br)cnn2C)C2(CCCC2)C1 c1(C(N2CCOCC(NC(c3ccc(Br)o3)=O)C2)=O)ccc(Cl)cc1[N+](=O)[O-] c1(C(=O)N)occ2c1CCOC2.C1(COCC(=O)NC2(CC)CCCC2)CCCOC1 Cn1c(O)nc(NC(C2CCC3C(C2)C3(F)F)=O)cc1=O c1(C(=O)NCC(CN(C(C2C(=C)C2)=O)C)(C)C)ccccc1C N1(C(CC=C)=O)CCC(C)(CNC(C2CCCN(CC)C2)=O)CC1 c1(C(=O)NC2C(NC(=O)Cc3ccc(CO)cc3)CCC2)cnc(O)cc1O N1(C(c2cc(C)nn2C)=O)C2CCC1C(CO)N(C(c1c(C)nn(C)c1C)=O)C2 CC(C)(C)C(C(=O)NCCCCNC(C1COC1)=O)C1CCCC1 c1(C(N2CC(F)(CNC(c3n(CC#C)ccc3)=O)C2)=O)ccc2c(c1)CCS2 c1(OC)cc(F)cc(C=CC(N2CC(C(=O)Nc3cc(F)ccc3F)C2)=O)c1 n1(C(C)C)ncc(C(=O)NC2CC(NC(C3(C)COCCO3)=O)C(O)C2)c1Cl CC(CC(=O)NC(C)(CNC(c1coc(Br)n1)=O)C1CC1)C1CCC1 C(CCC(=O)OC)(C(=O)NC(CC(C)C)C(=O)OC)N(C(C(=O)OCC)C)C c1(NC(CC2CN(C(C#CC(C)C)=O)C(C)(C)C2)=O)ccc2nonc2c1 C1(NC(C=C(C)Cl)=O)C(C)CCN(C(=O)CC23CCC(CC2)C3)C1C C1(C(=O)NC2CN(C(c3c(OC)nsc3)=O)CC2SC)C2CCC3C(C2)CC13 C1(NC2(C(=O)NC(C3CC3c3ccc(C)o3)=O)CCCC2)CCCC1(C)C C1(NC(C2(C=C)CCC2)=O)CC2(C1)CC2C(=O)NCCOC C(=O)(CCCCC(F)F)N1CCC(C)C(N(C)C(C2C(C)C2C)=O)C1 N1(c2n(CC(C)C)c(C3CCCS3)nn2)CC2C3CCC(C3)C2(CC)C1 CN1CCC(O)(CC(=O)NC2C3CCN(C(=O)CC4CC5(CC5)CO4)CC23)CC1 C1(C(=O)NCCC(=C)C)CCC(C(=O)NCC2(SCC)CC(=O)C2)CC1 Cc1cc(C(=O)NC(CO)C(=O)N(CCCC(F)(F)F)CCO)ccn1 C(=O)(C1CCc2nccn21)N(C(C1(C)CC1)C)C.C12CCN(C1)C2=O N1(C(CC2C(C)CCO2)=O)CCC(C(=O)NC2(C3CC3)CCOC2)=C(F)C1 C1(C(N(C)CC2CCSC2)=O)CCCC(NC(=O)C(C)(C)C2CCOC2)C1 N(C(=NCCCCC(F)(F)F)N1CCc2nnc(O)cc2C1)CC(C(C)C)(C)C c12ccc(cc1C)CCN2.c12ccc(nc1)CNC(=O)CCC21CC1.CO.OC c1(C(C(N2CCC(C(F)F)(CNC(CSCC)=O)C2)=O)C)c(C)nn(C)c1C c1(C(N2CCC(N(C(=O)Cc3cncnc3O)CCC)C2)=O)ccc(Cl)cc1Cl S(=O)(=O)(c1ccccc1Cl)NC1CN(C(c2c(C)cc(Cl)nc2Cl)=O)C1 C#CCC(C)(C)C(=O)NCC1C2CN(C(=O)Cc3c(Cl)cnn3C)CC12 C(CCCCC(F)(F)F)NC(C12CC(C(=O)Nc3c(C#N)ccs3)(C1)C2)=O c1(C(=O)NC(C(C)NC(CCCCC(C)C)=O)C)cnn2c1C(C)CCC2 c1(C(N2CCN(C(c3c(=N)[nH]c(C4CC4)nc3)=O)CC2)=O)noc2c1COCC2 Cc1ccc(CO)o1.N12CC(CO)(C1)C2=O.C(CCN=[N+]=[N-])OCCO c1(C(=O)NCCN(CC(C)O)C(N2CC(C(=O)N)C2)=O)cscc1C.N(C)C C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)C(NC(c2c(C)cns2)=O)C1C CCC(CCC(F)(F)F)(c1nnnn1C1CC1)NCCn1ccnc1 c1(C(=O)NCC=CCNC(C2C(C)N(C)CC2)=O)cccc2c1OCC2(C)C CC(C)C(CC(=O)NC12COCC(C1)C2)NC(=O)NC(C)(C)C N1(C(C=CC)=O)CCOC(CCNC(c2cccc(OC(F)F)n2)=O)C1 N1(CCC)CCC(N=c2[nH]c(=NC3CCN(C(C)=O)C3)c3c(ncn3C)[nH]2)C1 N1(C(C2(CNC(c3cc(CCC)on3)=O)CCCO2)=O)CCC2CC2C1 c1(C(=O)NC2CC(F)(CNC(c3c(CC#N)ccs3)=O)C2)ncc2ccccn12 C#Cc1cc(C(N2CCN(C(C3CCC(C(N)=O)CC3)=O)C3CC23)=O)ccc1C Cc1nc(N(C2CCS(=O)(=O)C2)CC2CCC2)cc(O)n1 C1(NC(C2CC3(CC(C)(C)C3)C2)=O)CCCC12CCOCC2 c1(C(=O)NCCO)ccccc1OCCN(CC=C)CCNC(=O)CSC(F)(F)F Cc1ccc(C(=O)N(C2CCC(NC(c3cn(C(F)F)cn3)=O)C2)C)nn1 c1(CC(=O)Nc2cc(N)cc(Br)n2)noc2ccc(Br)cc12 C(CC(=O)NCC1(O)CN(C)C1)(C(F)(F)F)NC(C(CC(C)C)OC)=O Cc1c[nH]cc(C(=O)NCC2CC2NC(c2cccc(C(F)(F)F)c2O)=O)c1=O N1(C(c2cnc(C)o2)=O)CCCCC(NC(=O)CC2CCC(C)C2)C1 CCC(CC(=O)NC1(C)CCN(C(C2CC3CCC(C2)N3CC)=O)CC1)C(F)F N(C1CC(C)n2ccnc21)C(C1=CCN(C(c2c(C)cc(C)o2)=O)C1)=O C1(CNC(=O)NCCN=c2cc(C3CCCC3)nc[nH]2)Cc2ccccc2CO1 C12(CNC(C(CC)NC(N)=O)=O)CN(C(c3cc(=O)cc[nH]3)=O)CC1CCO2 c12ncccc1CO2.C(CCC(=O)NCCCCNC(=O)OC(C)(C)C)OC c1(CC(=O)NC2CCC(F)(CNC(=O)CC3(CO)CC3)C2)coc2ccccc12 c1(NCC)cncc(C(=O)O)c1.C1(CN)CCC(CN)O1 N1(C(c2cc(C)on2)=O)CC2(CCN(C(=O)C(C)(C)CF)CC2)C1 N1(C(c2nccc(OC)n2)=O)CC2(C)CN(C(=O)C3CC3)CC2(C)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CC(F)(CNC(C2COCCOC2)=O)C1 c1(C(=O)NCC(C2CCCCC2)NC(CN2CC(C)C2)=O)noc2c1CCCC2 c1(C(N2CCC(CN(C(=O)CC34CCCC3C4)C)C2)=O)cc(F)c2[nH]nnc2c1 c1(C(C(CC)C)O)nc(CCC(C)C)nn1-c1ccc(Oc2ccccc2)cc1 C(=O)(C1=CCCCCC1)NC1CCC(N(C(=O)CCc2nnc(O)nc2O)C)C1 c1(C(=O)NC(C(CO)NC(C2(SC)CC2)=O)C)coc2c1NC(=O)CCC2 C1(NC(=O)C(O)Cc2ccccc2)CCN(C(C2CCCC3(CC3)C2)=O)CC1F CC(N=c1nc(N2CCCC(OCCO)C2)c2[nH]ccc2[nH]1)C(C)CO C(=O)(C(C)(C)Nc1ccccc1)NCC(C)NC(=O)C(O)Cc1cnc[nH]1 C(=O)(CN=c1nc(-c2cc(F)cc(F)c2)[nH][nH]1)NC(c1n(C)cnn1)C(C)(C)C c1(NC(C23C(CN(C(c4cnco4)=O)C2)C3)=O)nc(Cl)cnc1Cl CCC(CCCC(=O)N(C1CC(=C)C1)C)NC(=O)CC1CCCCO1 N1(C(c2cnc(CCC)s2)=O)CCCC1(C)CCCNC(=O)C=C(C)C C12(C(=O)NCC3N(C(CC4(C)CCCCC4)=O)CC3)CCCC(C1)C(=O)NC2 N1(C(c2ccc(C#N)s2)=O)CC2CCC(C1)N2Cc1cccc2occc12 Cc1nc(CCC(=O)NCC2(F)CCN(C(=O)C=Cc3ccccc3)C2)[nH]c1C c1(C(=O)NCCC2(NC(C(N3CCN(C)CC3)C)=O)CC2)ccnc2[nH]nnc12 N1(C(CC(=C)C)=O)CCN2C(=O)C(NC(c3ccc(CC(C)C)s3)=O)CC2C1 CC(CS(C)(=O)=O)C(=O)NC1CCN(C(C2CCC23CCC3)=O)CC1 c1(C(N(CCC)CCNC(=O)Cc2csc(C)n2)=O)cnn2c1CN(C)CC2 C1(C(=O)NCC(=O)NC2CCC2)CC2(CCN1C(=O)C(F)C(F)(F)F)CC2 c1(C(=O)NC(CN(C(c2nnc(S)n2C)=O)CC)C)cc(F)cc(S(N)(=O)=O)c1 C1(NC(C2N(CCC)CCC2)=O)CC(NC(c2oc(C(C)C)nc2C)=O)CC1O C1(NC(c2cc(C)ncn2)=O)CC2(C1)CC(NC(=O)CN1CCC(C)(C)C1)C2 Cc1nc(O)sc1C(N1CCC(O)(CN(C(=O)Cc2cc(C)n(C)n2)C)C1)=O CN1CCCCC12CN(C(C1CC(NC(C3(C)CC3)=O)CCO1)=O)C2 C1(CN(C(C(C)Cc2cnc[nH]2)=O)C)CC(F)CN1C(=O)C(c1ccn(C)n1)C c1(OC)nc(C)ccc1-c1ccc(C(=O)NCc2ccc(O)c(C)c2)nc1 c1(CC(=O)NC2CN(C(CC(C)(C)C)=O)C3C2C3)ccc2c(c1)OCO2 CCC(CN(C)C)C(=O)NC(c1cccnc1)C(N1CCCC1C1CCOC1)=O N1(C(c2scc(C)c2)=O)CCC(OCc2cn(CC3CC3)nn2)CC1 C1(NCCNCCOC)(CO)CCC2CCCC12 N#CC(=O)C(CC(=O)CC1CCCCC1=O)(F)c1ccccc1.OCN c1(NC)cncc(C(=O)OC)c1.c12nnnn1CC2(C)NCCCCC C1(C(=O)NCc2nn(C)c(=O)o2)(OC)CCN(C(=O)CN2CCC(=O)CC2)C1 c1(NC(c2c(OC)cccc2)(C)C)cccc(S(=O)(=O)NC2CC3CC3C2)n1 n1(CCC(=O)N(C(C)C(C)C)CCOC)cc(-c2ccnn2-c2ccccc2)nn1 O=C1CC2(CCN(C(c3cc4cccc(-c5ccc(F)nc5)c4s3)=O)CC2)CN1 C(C(CC1CC1)C(=O)NC(c1n[nH]c(C)n1)CO)NC(C(CC)C)=O C1(CNC(CCC=C)=O)CN(C(c2ccsc2Cl)=O)C(C)(C)C1 C1(NCc2ccc(Cl)cc2)CN(C(=O)Cc2c(Cl)cccc2Cl)CCN1OC C1(CNC(c2c(CC)scc2)=O)CCC2(CN(C(c3cnn[nH]3)=O)C2)O1 C12C3CN(CC13)C(=O)C1(CC1)NC2=O.N1(CCSc2ccccc2)CC2CC2C1 c1(CC(=O)NC2C(CNC(c3c(CC)scn3)=O)C2)ccc(C)nc1 C1(SCC(N2CCCC(OC(=O)COC)C2=O)=O)CC2(C1)C(F)(F)C21CCC1 C1(CCC)(C(=O)NCCN2CCN(C(C3CCCOCC3)=O)CC2)CCNC1=O C(=O)(CC(O)C(Cl)(Cl)Cl)NC(=O)CCCCc1cn(C(CC)CC)nn1 c1(OC)cccc(N=CCC2(S(=O)(=O)NCc3nc(C(C)C)no3)CCC2)c1F N1(C(c2cc(C)[nH]n2)=O)CC(C(=O)N(C(C)C(C)(C)C)C)C2(CCC2)C1 c1(C(N(C2CCN(C(c3ocnc3C3CC3)=O)CC2)C)=O)onc2ccccc12 CC1=C(C(=O)NCC2CC(C)N(C(C3CC3c3ccc(Cl)cc3)=O)C2)CCC1 c1(C(=O)NCC23N(C(COC(C)=O)=O)CC(CO)(C2)C3)ccc2cc(C)cn2c1 N1(C(C2(C)CCC2)=O)CC2CCCC2(CNC(=O)Cc2ccc3c[nH]nc3c2)C1 Cn1cnc(C(N2CCCCCC2C(=O)NCCCCCCC2CC2)=O)cc1=O Cc1c(Cl)sc(Cl)c1C(N1C(CNC(=O)C(C)CN(C)C)CC2CC12)=O N1(C(C(COC)OC)=O)CC2C(NC(=O)Cc3ccc(OC)nc3)C2C1 c1(C(=O)NCCCN(C(c2c(C)ncn2O)=O)CC)coc2c1CS(=O)(=O)C2 c1(CC(=O)NCC(CN(C(C(CC)O)=O)C)C)ccccc1SC(C)C(N)=O c1(Cn2c(N3CCOC(C)C3)nnc2COC2CCOC2)cnc(O)nc1O C=CCC(CC(C)C)C(=O)NCCn1cc(C(=O)NC2CC2CC(C)(C)C)nn1 c1(OCC)ccc(S(=O)(=O)N(C2CCCCCC2)C)c2ncccc12 c1(C(C#C)C)nnc(N2CCN(C)CC2)n1Cc1cccc(OC)c1 c1(C(=O)NCCCC(CCC)NC(=O)CCC(C)SC)cc2nc(F)ccc2o1 CCC(C)C(C)(O)CNC(=O)C(Cc1cc[nH]n1)NC(=O)C(C)c1cccs1 CC1(C)CC(CC(=O)NCCC2CN(C(C34CCCC3CCC4)=O)C2)C(C)(C)O1 c1(OC)cncc(C(N2CC(F)(CNC(=O)C=C(C)CN3CCCCC3)C2)=O)n1 CC(C)(C)CC(O)C(=O)N1CCN(C(=O)C=Cc2ccc(C(N)=O)o2)CC1 c1(C(=O)NC2CCC(NC(c3nccc(OC)c3)=O)C2)c(OC)ccc(Cl)c1F C1(NC(c2cccc(OC(C)C)c2)=O)CN(C(c2nnn(C)c2N)=O)CC12CC2 C=C(CNC(C1CCN(C(=O)CS(C)(=O)=O)C(C)C1)=O)C(F)(F)F C=CC(C)(C)CC(=O)NCCC(C)NC(c1cccc(C(N)=O)c1)=O N1(CC(=O)N(C(C(=O)N(CC(CCC)O)C)C)C)CCC(C)CC1 N1(C(CCCNC(C)=O)=O)CC2(CC(NC(=O)C3CC3)CO2)C1 c1(C(=O)NC(CC)CNC(c2cc(F)c(OC)cc2N)=O)ccc(Cl)c(C)c1N N12CCC(C)(C1)C(=O)NCCC2=O.C1(CC(=O)NC2C(C)C2)CCCCC1 C1(C(NC[Si](C)(C)C)=O)CC2CCCC2N1C(c1ncc2ccccn12)=O N1(C(c2ccc(Br)c(C)c2)C(=O)NCC)CCCC1(C)P(C)(C)=O N1(C(c2c(C)csc2)=O)CCC2CC(C1)CN(C(=O)CS(C)(=O)=O)C2 C1(NC(c2c(C)nc3ccccn32)=O)CCOC12CCN(C(=O)CC(C)C)CC2 c1(OCC)cc(C(=O)NC(C2CCCN2C(C2C(C)C2C)=O)C)ccc1C c1(C(=O)NC2CCCCC2CNCC2CC(C(F)(F)F)CO2)c(F)ccc(Cl)c1F Cn1ncc(C(=O)NC2CCCC(NC(C3(O)CCC3)=O)C2)c1C(F)F Cc1nc(NC2CC(NC(c3ccc(F)c(Cl)c3F)=O)C2)c(Cl)cc1C#N N1(C(CC=CCC)=O)CCCCC1C(=O)NCC1(CC(C)C)CC1 CCC(C)C(O)C(=O)NCC(c1ccc(C)cc1)NC(c1cc2occc2[nH]1)=O N1(C(=O)Nc2cn(CC=C)nc2)CCC(CNC(C)=O)CC1 C1(CNC(C(COCC)n2cc(CCc3cc[nH]n3)nn2)=O)C2C3CCC(C3)C12 C(=O)(CC(C)C(=O)NCC12CC1CN(C(=O)C1=CCCCC1)C2)OC c1(C(=O)OC)cccc(CO)n1.n1(CC)cc(C(C)N(C)C(=O)N)nn1 C1(CC(=O)NCC2CCCN2C(c2nnsc2-c2ccccc2)=O)COCCO1 CCC(CC)C(C(=O)NCC(O)CNC(c1cnc(O)cc1C)=O)OC C=C(C)CC(C(=O)NCc1ccsc1C(=O)NCCc1c[nH]nc1O)OC C(CNC(=O)CC1OCCCO1)(C(=O)NCC1(n2cccn2)CC1)N(C)C N1(C(C2C(C)OCCC2)=O)CCc2nc(O)cc(C(=O)NCC(F)C3CCC3)c2C1 CN1CCCC1C=CC(=O)NCC=CCNC(c1csc(C(F)(F)F)c1)=O c1(CC)cc(N2CC(NC(=O)COC(C)CC)C(C)C2)nc(C)n1.C1CO1 c1(CC)cc(C(=O)N(C(c2ccccc2)CNC(=O)C(CC)SC)C)cc(F)c1 N1(C(C=Cc2ccc(CC)o2)=O)CCC(NC(=O)Cn2cccc2)C(O)C1 C1(C(=O)NC(c2csc(CCC3CCCNC3)n2)C)CCc2nc(=N)[nH]cc2C1 C(=O)(CC(=O)N(CC(O)CNC(c1cc(F)c[nH]1)=O)C)NCC C1(NC(c2cnc(O)cc2O)=O)CN(C(=O)Cn2cccnc2=O)CCC1CO c1(C(N(C(CN(C(C(C=CC)O)=O)C)C)C)=O)c(C)coc1C(C)(C)C N1(C(c2c(C)onc2Br)=O)CC(NC(C2C=CCC2)=O)C2(CC2)C1 N1(c2c(C(=O)OC)ccc(O)n2)CCC2(CCCCN(C(c3ccoc3)=O)C2)C1 C1N=C2C=C(N=CN2)NCC2CCCC12.c1(C(C)C)nccn1C(C)(C)C Cc1cc(C#N)ccc1C(N1CC(O)CC1(C)C(N1CC2(C1)CC2(F)F)=O)=O C(=O)(CCCCC(C)=O)N1C(C(N(CCCCC)C(C)C)=O)CCC12CC2 c1(CC(N2CCC(CNC(=O)CC3CCOC3)C2)=O)ccc(Br)c(Cl)c1 C(=O)(C(C)(C)C(C)(C)O)NC(c1ccccc1)C(=O)NC(C1CCCCC1)C#C c1(CC)nc(C)[nH]c1C(=O)NCC1CN(C(c2ocnc2C(F)(F)F)=O)CC1C CC1C2CCC(C2)C1C(N1CCCCC1C1CCN(C(C2CCSCC2)=O)C1)=O C1(C(N2CC(N(C)C(c3nonc3N)=O)C2)=O)CC2CCCC12 C1(C(=O)NC(CCF)C(=O)OC)(CC)CCN(C(C2CC3CCCC3C2)=O)CC1 N1(C(C(C=C=C)C)=O)CCn2nc(CNC(=O)CCNC(N)=O)cc2C1 c1(CC(=O)OCCc2ccco2)cccc(CCF)c1 C(CC(C)C)(C(=O)NC1CC1O)NC(CCOCCC)=O Cc1c(F)cc(NC(C2CC(F)CN2C(c2cc(Br)ccc2Cl)=O)=O)cc1Br CC(C)C(CN(C)C)C(=O)NC(C)(C(N1CCOC2CC12)=O)C1CC1 C1(CC)CCN(C(c2c[nH]c(=O)cn2)=O)C1CNC(c1ccc(OC)nc1)=O C=C(C)c1ccccc1NC(C1CCCN(c2ccnc3ccnn23)C1)=O C1(CC=C)(NC(=O)C(c2cccc(F)c2)C)CCCN(C(=O)C(C)(C)C(C)C)C1 CCCCCC(F)C(=O)N(C(C)C(=O)NCC1CCCC2(CC2)C1)CC CC1(C)CCCC(C(N2CCC(F)(CNC(=O)CC3COCCO3)CC2)=O)C1 C(=O)(CCC(=O)c1cc(Cl)sc1Cl)N1CC(NC(C2(CC#C)CC2)=O)C1 C(=O)(C(F)CC(CC)CC)N1CC(NC(CCCC)=O)C(O)C1 c1(C(N2CCC(N(CC)Cc3onc(CC)n3)CC2)=O)ccc2c(c1)COC2 N1(C(=O)Cc2ccon2)CCC(C2CCCN(C(C3(CCCF)CC3)=O)C2)C1 C(=O)(C1CCc2cccc(OC)c21)N1C(CNC(c2cncc(C=C)c2)=O)CCC1 c1(C(N2CC(NC(CC(C)c3ccco3)=O)(CO)C2)=O)cccc2c1OCC2 c1(SC2(C(=O)NC3CC(N(C(C4C(C)C4C)=O)C)C3)CC2)ccccc1 N1(C(C=Cc2c(C)cncc2)=O)CC(NC(=O)Cc2nocc2C)C2(CCC2)C1 c1(C(=O)NC2(CC)CCN(C(C(CC)C)=O)CC2)cccc2c1CCCC2=O CC(CC(=O)NOCC(=O)NC(C)C(=O)NC1CC1)N(C)C.C(C1CC1)N Cc1nc(CNC(C2(O)CCSC2)C)sc1C Cn1cc(Cl)cc1C(=O)N(CCCNC(=O)COC1CC=CC1)CC1CCCC1 C(=O)(CC(C)(C)CNC(C1(C)CCCCC1C)=O)N(C)Cc1n(CC)cnn1 N1(C(C2C3(CCN(C(CC4(C)CCOC4)=O)C3)C2)=O)CCCC2(CC1)CC2 c1(C(C(=O)N(c2c(C)n[nH]c2)C2CCCC2)O)ccc(C(C)C)cc1 C1(C(=O)NC(C2C(C(=O)OC)C2)=O)CCN(C(c2onc(OC)c2Br)=O)CC1O CCCC1C(=O)NCCC(OC)CNC(=O)C2(CC2)C(=O)N1.C1(CC)CCC1 C1(NC(C=CCOC)=O)CN(C(c2ccc(F)c(F)c2C)=O)CC12CCC2 C(C(CC(C)C)C(=O)NC1CC(C)(C)C1)NC(C1(CCCC)CCC1)=O Cc1cc(NCC(C2CC2)NC(C2COCCN2C)=O)n2ncnc2n1 Cc1[nH]nc(Cl)c1C(=O)NCC1C2CN(c3cc(C(F)F)ncn3)CC12 c1(C(=O)OC)n[nH]c2cc(CNC(=O)NC3CC4OC3C3CC43)ccc12 c1(C(N2CC(NC(C(CC#C)C)=O)CC2(C)C)=O)cc2cc(C)ccc2[nH]1 c1(CC)ccc(CCCC(=O)NC2CN(Cc3csc(=N)[nH]3)C2)cc1 c1(C(C)C)nnsc1NCCC(Cc1ccccc1)NC(=O)OC(C)(C)C Cc1ccnc(C(N2CCC(C)(C(=O)N(C)CC3CCCC4CC34)C2)=O)c1 c1(C(CNC(C(C2CCOC2)OCC)=O)C)ccc(F)c(F)c1 C1(C(N)=O)CN(C(=O)Cc2cnnn2C)CCC1NC(=O)CN1CCOCC1=O c1(CN2C(C)(C(=O)Nc3cocn3)CC2)cc(Br)ccc1O N1(C(C2N(C)CCN(C(c3c(C)cc(F)cc3)=O)C2)=O)CC2CC(C)(C)C2C1 C1(C(=O)NCC(C)(C2CC2)NC(C2CCSCC2)=O)OC2CCC1C2 c1(C(N2CCCN(C(CCC(=C)Cl)=O)CCC2)=O)cc2c(o1)CCCNC2=O N1(C(C=CC=CC)=O)CC(CNC(=O)C=Cc2cccc(CO)c2)CC12CCC2 CN1CCN(C(=O)CC=Cc2ccccc2F)C(CNC(C2CCCS2)=O)C1 c1(C(=O)NCC2CCN(C(c3cn(CC=C)nn3)=O)C2)ccc(Cl)c(O)c1 C1(=O)CC(C)(C)CN1.C(C(C)(C)C(=O)NC(C)CC1CCCCC1)OC.C(C)(C)(C)O c1(C(=O)NCC(C)NC(C(CCC)CC)=O)snc2ccc(Br)cc12 CC1CCN(Cc2csc3cc(Br)ccc23)CC2(CCOC2)O1 CCC(CC)CCC(=O)N(CC(C)CNC(c1ccc(Cl)c(F)c1F)=O)C C1(C(F)(F)F)CC2CCC1C2.C1(CNC)OCCC1(C)C Cc1ccc(CC(=O)NCC2CCCN2C(=O)C(C)n2cccc2)c(Cl)n1 c1(C(N2CC3CC(NC(CSCC(C)=O)=O)C3C2)=O)cc2c(C)cccn2c1 CC1CN(C(=O)C#CC2CC2)CC1NC(=O)C(F)(F)Cc1ccccc1 Cc1cccc2c1CCOC2C(=O)NC(C)C(C)NC(=O)Cn1cncn1 c1(CC(C(=O)NCc2cccnn2)NC(CC(CC)OC)=O)ccc(Cl)cc1Cl N1(C(C(=O)NCCOC)=O)CCC(N(C)C(c2cc(COC)n(C)n2)=O)CC1 c1(C(=O)NCC(C)NC(C2CC2C(N)=O)=O)ccc(N)c2ccncc12 c1(C(=O)NC(C2CCCN(C(=O)OCC)C2)C)cc2c(s1)COCC2 C(=O)(C(C)(C)C(C)(C)C)N1CC(OC)C(NC(=O)C(c2cccc(F)c2)O)CC1 c1(CN2CCC(NC(c3ccc(C(=O)OC)s3)=O)CC2)ccc(N(C)C)c(Cl)c1 C(CN=c1[nH]c(N2CCN(CC)C(=O)C2)nc2c1COC2)N1CCC(OCC)C1 C(=O)(C1CCC(=O)c2cccn21)N(CCCN(C)C(c1ccc(C(F)F)o1)=O)C Cc1cccc(C(O)C(N2CCC(O)(CCNC(=O)CC=C(Cl)Cl)C2)=O)c1 c1(C(=O)NC2CC(C)(NC(C3C(C)CC3)=O)C2)ccc(N)cc1Br c1(NC(c2c(CNC(C(CC=C)(C)O)=O)ccs2)=O)cccc(C)c1C#N N1(C(c2noc(CC)c2C)=O)CCCC(C)(NC(=O)C(N2CCC(C)(O)C2)=O)C1 c1(CC(=O)NC2CCN(C(CO)=O)C2)ccc(Cl)cc1.Cc1cc(NC2CC2)no1 c1(NC(=O)NCC2CCN(Cc3ccccc3)C2)nnc2n1CCCC2 c1(C(=O)NCCCN(C(C2C=CC=CC=C2)=O)CC)cccc2ccoc12 C1(NC(CN2C(C)CCC2C)=O)CCN(Cc2ccccc2C(F)(F)F)C(C)C1 c1(OCC)nccc(C(N2CCC(N(C)Cc3ncc(Br)cc3F)C2)=O)c1Cl c1(OC)ncc(F)cc1C(=O)NC1CCCC1C(N1CCCC(C)CC1)=O N1(CC(=O)NCC(CC)(C)NC(=O)C(F)OC)CCNC(=O)C1 C(C(C(=O)NCC1(NC(c2nc(C(N)=O)no2)=O)CCC1)N(C)C)OC CC(O)C(C(=O)NCc1cc(C(=O)NCC2CCSC2)co1)N(C)C c1(NC(C(C(C)C)C)CNC(C2(CF)CC2)=O)nc2ncc(Cl)cc2s1 C(=O)(C1=NOC(C)C1)N1CC(C#C)(C(N2CCN(C(=O)CO)CC2)=O)C1 N1(C(CN(CC)CC)=O)CCC(NC(=O)CCN2CCCCC2)C(F)C1 C1(c2nnnn2C2COC2)(NC2CCC(COC)CC2)CC2(CCCCC2)C1 N1(C(CCC=C)=O)CCCC(N(CCF)C(c2sc(C)cc2C)=O)C1 N1(CCOCC)CC(C2CCCN(C(=O)C(C)(F)F)C2)C1 N1(C(CC(C(C)C)NC(=O)CCC2CC2)=O)CCC2CCCC2CC1 c1(C(N2CCN(CC(N)=O)CC2)C(=O)NCCOCC)cnn(CCO)c1Cl.CC c1(C(N2CCN(C(CCC(=C)Cl)=O)C(CC)C2)=O)cc(C)c2ncccc2c1 S(=O)(=O)(c1cccc(Br)c1)N1Cc2c(cccc2)C1.C1(CC(N)=O)CCCCN1 CCN(NC(=O)CCc1nc(CN)n[nH]1)S(=O)(=O)CC.C1(OC=O)CCS(=O)(=O)CC1 C=CC(C)CC(=O)N1CC(O)CC1C(N1CCOC(CC)C1)=O N1(C(C2N(C)CCOC2)=O)CCN(C(c2ccccc2CO)=O)CC1CCO C1(NC(c2cc(CCOC)on2)=O)CN(C(=O)C=C(C)Cl)CC1CC1CC1 C1(NC(C2(NC(=O)NC)CCCC2)=O)CN(C(c2[nH]nnc2C)=O)C2CC12 N1(C(CC(C)(C)O)=O)CC2CN(C(=O)CNC(c3ccc(Br)o3)=O)CCC12 c1(OC)nc(N2CC3C(C2)N3C(c2ccc(OC(F)F)cc2)=O)ncc1C#N C1(C#N)(C(=O)NCC2CCC(NC(CC)=O)C2)CCCO1 c1(C(=O)NCC2(O)CN(C(C(CCC)N(C)C)=O)C2)[nH]cc2c1CCC2 Cn1cncc1C(O)C(=O)NC(C1CCN(C(=O)C(C)(C)C)C1)(C)C C(=O)(CCC(C)C)NCC(CNC(c1nc(COC)sc1)=O)(C)F C1(N)(CC(=O)N(C2CCN(c3ccccc3)C2)CC)CCOCC1 CC1=C(C(=O)NC2CC2CNC(C2CC(Cc3cccnc3)C2)=O)CCCC1 c1(CNC2C(C(N3CCN(CC#C)CC3)=O)CCCC2)ccc([N+](=O)[O-])cc1F Cc1c(C(=O)N(C)CCN(C)C(C2C3CCC(C3)C2(C)C)=O)oc2ccccc12 C=CC(CC)C(=O)NC1COCC1NC(=O)CCCN1C(=O)CNC1=O CCCS(=O)(=O)CC(=O)N1CCC(CN(C)C(c2ccn3nnnc3c2)=O)C1 C1(CNC(=O)Cc2cnc[nH]2)CN(C(=O)CNC(=O)NC2CC2)CC1O C(C(=O)NCc1cccs1)(C(C)CC1CC1)N1C(C(=O)OC)CN(C)CC1 Cc1ccc(C(=O)NCC2CCCN2C(=O)CC2CCCC(C)(C)O2)c(F)c1C C1(N(C(=O)C(=O)NC2CC(C)C2)C)CCN(C(=O)CCSC2CC2)CC(C)(C)C1 c1(C(C2CCCOC2)N(C(=O)NCC2C(C)C2)C)ccc(F)c(F)c1 C(=O)(C1=COCC1)NC(C(=O)N(C(CCC)C)C)C1(O)CCC1 C1(NC(CC2CCN(C(C3(COC)CC=CC3)=O)CC2)=O)CC2C(C1)C2(F)F c1(OCC(=O)N(C2CCC(CC3CCC3)CC2)C)c(F)cccc1[N+](=O)[O-] N1(C(C)C)CCOC(C(=O)NCc2cccc(CNC(=O)C(O)C(F)F)c2)C1 C1(C(N2CC(F)CC(NC(Cc3c(C)cco3)=O)C2)=O)CC2CCCC(C1)C2 C1(CCC)CN(C(C2CC23CCC3)=O)CCN1C(c1cnc(NC(C)=O)o1)=O CC1CCn2cc(C(=O)NC3CCN(C(C4C(C)(C)C4(C)C)=O)CC3O)nc2C1 CC1COCC(CC(=O)NCC2(C(=O)NCCCCF)CC=CC2)O1 CC(C)C(F)(CNC(=O)CCN(C)C)C(=O)N1CC2(CCOC2)C1 C(=O)(C1CCC2(CN(C(=O)Cc3cccc(C(F)(F)F)n3)C2)OC1)OCC CC(C)C(C)C(=O)Nc1cccc(CNC(=O)CC2(C)CCCO2)c1 c1(CCNC(c2c(CNC(c3csc(Cl)n3)=O)n[nH]c2)=O)cccc(F)n1 c1(C(N2CCN(C(C(OC)OC)=O)C(C#N)C2)=O)ccc(Br)c2cccnc12 Nc1ccc(C(N2CCCN(C(c3cnns3)=O)CC2)=O)c2cnccc12 Cn1c2nnc1CSC2c1nnnn1CCCF.c1(C)cnc(C(F)F)s1.C(CO)O c1(C(=O)NC2CC(OC)CN(C(=O)C3CC3)C2)cc2n(n1)CCCC2O N1(C(C2(C)C=CCC2)=O)CCC(C)(C(F)C(=O)NCCN(C)C2CC2)C1 c1(C(=O)NC2CC(F)(CNC(C3CC(C)CC(C)C3)=O)C2)ncc2n1CCCC2 n1(CC(=O)NC2C(CNC(C3(N(C)C)CCCOC3)=O)C2)ccc([N+](=O)[O-])n1 C1(C(=O)NCC(C)N(C)C(C2CCCCN(C)C2=O)=O)CCN(S(N)(=O)=O)CC1 Cc1ccc(F)c2oc(C(=O)NCCOCCN(C)C(C3CCCSS3)=O)cc12 N1(C(CCCC(C)=O)=O)CC=C(CCNC(C2(C)CCN(C)C2=O)=O)CC1 c1(C(C)NC(C(CCCC)(F)F)=O)ccc2c(c1)CN(C(=O)C(C)OCC)C2 N1(CC)CC(C(N2CCCC2NC(=O)C(C)(C)C#N)=O)CC1=O c1(CC)ccc(C)cc1C(=O)NCC1CCCN(C(C2CC(C)C2)=O)C1 C(=O)(C(O)C1=CCCCC1)N1CC2C(CNC(C3CC3[N+](=O)[O-])=O)C(CC2)C1 c1(OC)cc(C)sc1C(=O)NCCN1CC(c2ccc(F)cc2)CC1=O c1(-c2ccc(C(=O)OCC)s2)cc(C)[nH]c1C.c1(N)cc(OC)nc(OC)c1.SC N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(c2cc(N)ccc2F)=O)CC1C(F)F Cc1cc(=NC(CNC(C23CC4CC(C2)CC(C)(C4)C3)=O)CO)[nH]c(C(C)C)n1 C=CCC(C)(O)C(=O)NCC1CC1CC(N1C2CCC1COC2)=O C=C=CCCN=c1[nH]c(N2CCC(N(C(=O)NC)C3CC3)CC2)nc2ccsc12 C(=O)(C1=CC2CCC(C1)C2)NC1C2N(C(C(=O)NC(C)C)=O)CC(CC2)C1 c1(N(C)CC2CCN(C(c3c(C(C)C)cccc3)=O)C2)ncc2c(n1)CCCC2 C1(NC(CC(C)N(C)C)=O)CN(C(c2cc3ccsc3s2)=O)CC1(C)C N1(C(C(C2CC2)OC)=O)CCC2(CCC(NC(=O)CSC(=N)N)CC2)C1 CC(=O)CCCC(=O)NC(CNC(c1scc(C)c1Cl)=O)C1CCC1 c1(C(N2CCN(C(CC3(CS(C)(=O)=O)CC3)=O)C3C2C3)=O)cc2c[nH]cnc-2n1 C12COC3CN(CC13)C2=O.n1(-c2ccccc2)ccc(NC(C2CC2(F)Cl)=O)n1 CC(C)C(C)(CNC(C1C2CCCC12)=O)NC(c1c(C(F)(F)F)ncn1O)=O c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)CCSC2)=O)nc(Cl)ccc1Br c1(C(=O)NC2C(NC(c3nc(C)nn3C)=O)C2)nc(C)c(C)nc1C c1(C(=O)NC2CC(CNC(C(C)SCC)=O)C2)ccc(Cl)nc1O c1(C(N2CC3C(CNC(C4CCC(F)(F)C4)=O)(C3)C2)=O)cc2c(o1)CCCNC2 C1(NC(C2(SC)CN(C(=O)NC(C)C(=O)NC)C2)=O)CCS(=O)(=O)C1.CO C1(C(N2CCC(CNC(C(CN(C)C)(C)C)=O)(CO)C2)=O)CC2OC(=O)OC2C1 N1(C(Cc2ccn(CC)n2)=O)CCOC(CN(C)C(C2(Cl)CC2(F)F)=O)C1 c1(C(C)OCC)nc(C(=O)N(CCNC(=O)C(C)(C)C2CCCC2)CC)co1.OCO C(C[Si](C)(C)C)NC(C(C)N(C)C(c1ncc[nH]1)=O)=O N(C1CCOc2ccccc21)(CC(C)Cc1ccc(F)cc1)CC N1(C(C2(CCOC)CC2)=O)CCCC(O)(CNC(c2cc(Br)c[nH]2)=O)C1 N1(C(=O)Cc2cc[nH]n2)CC2CC(NC(C3(CO)CCC3)=O)CC2C1 CN1CC(NC(=O)CSCCNC(C2CCC(=O)CC2C)=O)C2(CC2)C1=O C12(CNC(C)=O)COC(C(=O)Nc3c(Cc4ccccn4)noc3C)(C1)C2 C1(CNC(CCCCNC(C)=O)=O)CCN(C(c2conc2C(C)C)=O)CC1C C(=O)(CCCC(=O)C1CCCN1C(=O)OC(C)(C)C)OC(c1c(C)noc1C)=O C1(N(C(=O)CCNS(C)(=O)=O)C)CCCN(C(C2CC2C#N)=O)CC1 c1(C(=O)NCC2CN(C(=O)Cc3csc(Cl)c3)C2)cn2cccc(Cl)c2n1 N1(C(C(CO)NC(c2cc(CC3CC3)on2)=O)=O)CC(O)CC(O)C1 C1(C2C(N)C2)CCCC1(C)O.C(C(=O)NC1CC1NC(C1CCC1)=O)(OCC)OCC c1(C(N(CCCNC(=O)C(C2CC2)OCC)CC)=O)[nH]c2ccc(F)cc2c1Cl Cc1ccc2cc(C(=O)NC3CCCCCC3NC(c3ccc(Cl)s3)=O)cn2c1 C1(N(C(C(C)OCCC=C)=O)C)CCN(C(c2csnn2)=O)CC12CC2 C(=O)(CC(C=C)CCC)N1CCCN(C(CCC=C=C)=O)CC1 N1(C(C2C(=O)OCC2)=O)C2CCCC1CN(C(C1CN3CCN1CC3)=O)C2 c1(OCC(=O)NCC(C(C)C)CNC(C(C)OCC=C)=O)cccc(F)n1 CCCC(C(=O)NCCCC(C)NC(c1ccc(OC)s1)=O)S(N)(=O)=O c1(OC)ncccc1C(=O)NCCOCC(=O)NCc1ncn(C2CC2)n1 N1(C(C2(C)C=CCCC2)=O)CC2(CCNC(c3ccc(C(N)=O)s3)=O)CCC1C2 Cc1nc2ccccc2n1CC(=O)NCCCC1CCO1 N#Cc1cncnc1NC1CC1C(=O)Nc1cccc(CCO)c1 c1(NC2(c3n(CCCSC)nnn3)CCC2CC(C)C)cc(F)cnc1C#N C1(C(=O)OC)CSCN1C(=O)Cc1cn(CC2CCCCC2)nn1 C(=O)(CC(C)C(C)C)N(c1c(C)nc(C)[nH]1)CCO.n12cc(nn1)C21CC1 C1(C(=O)NCCCN(C(C=C(CC)CC2CCCCC2)=O)C)CCOC1C(C)C c1(C(N2C(CCCNC(c3c(C)c[nH]n3)=O)CCC2)=O)ccc(N)cc1Cl c1(OCC)ccc(OC2CCC2C(=O)NCC2CCCCC2)cc1C C1(NC(C(n2cc(C(CSCC)O)nn2)COC(C)C)=O)CCC(=O)CC1(C)C c1(NC(N(C)CCOCCN(C)C(C2(C)CC=CCC2)=O)=O)cc(N)ccc1O C=C(Cl)CC(C(=O)N(C)CC12CC(C1)C2)NC(=O)COCCC N1(C(C(=O)NC2CC(CCOC)C2)c2nc[nH]n2)CCC(O)C(C)C1 Cc1sc(S(=O)(=O)N2CCNC(CF)C2)cc1Br Cc1cccc(C(=O)C(N2CCCC(N(C)C(c3cc(CO)oc3C)=O)C2)=O)c1 C1(C(N2CCOC(C(=O)NC(c3ccc(O)nc3)C)C2)=O)(CC)CNC(=O)C1 CC(=O)C(C)(C)CC(=O)NC(CN=[N+]=[N-])C(=O)N1CCC(F)(CF)CC1 c1(NC(C23C(CN(C(C4CCCN4C4CC4)=O)C2)C3)C2CC2)c(O)cccc1Cl C(=O)(C(CCOC)OC)NC1(CC)CN(C(=O)CC2CC2C(F)(F)F)C1 C(CN=c1ccnc(N2CCC(C(C)C)C2)[nH]1)c1ccc(NC(CCC)=O)cc1 c1(N2CCCC(NC(C(CC)N(C)C)=O)C2)ncc(Br)c(O)n1 C12(C(=O)NCCOC3CCN(C(c4c(NC)cccn4)=O)C3)CC(C1)C(C)(C)O2 c1(-c2cc(C(=O)NCC3CC(NC(C4(C)CC4F)=O)C3)on2)ccccc1F C1(CC(N2CC(N(C(C(=O)OCC)=O)C3CC3)(CO)C2)=O)CCC(C)(C)O1 C1(C(N(c2cccc(Br)c2)C(CCC2(C)CCN2)=O)=O)CCCN(CC(F)F)C1 C(=O)(C(=O)N)NCCN(CC(C)O)CCSCC=C.C(COCCC1CC1)O c1(NC(c2c(SC)cccc2)C)ccc(S(=O)(=O)NCC2CCCOC2)cc1Cl N1(C(CC2C(OC)CC2)=O)CCC(C(C)NC(=O)CC(=O)N(C)C)CC1 C1(CNC(C(C)OCC)=O)CN(C(c2ncccc2Cl)=O)CCC1C CCC(CC)CCO.c12ccc(C)c(n1)ON(C1CCCC1)C2C(=O)NC C1(C(N(C)Cc2cn(CC3COCCO3)nn2)=O)CCCCS1(=O)=O C1(CNC(=O)CC2CC(F)C2)CCC(NC(c2occc2Cl)=O)CC1 c1(OC)ccc(CC(=O)NCC(CO)NC(C2CC2c2cccs2)=O)cn1 C1(NC(C(c2cccc(OC)c2)(F)F)=O)CCN(C(=O)Cn2ncnn2)CC1F c1(C(N(C(CN(C(C(COCC)C)=O)C)C)C)=O)cc(S(N)(=O)=O)cs1 CC(Cc1ccccn1)C(=O)N(C)CC1(O)CN(C(=O)C=C(Cl)Cl)C1 n1(CC)ccc(C(=O)NC(C(=O)NC(C23CC(CO2)C3)C)C2CC2)n1 c1(C(=O)NCC(=O)NC2CC2)cc2c(-c3ccc(O)c([N+](=O)[O-])c3)cccc2[nH]1 c1(CC(=O)NC23C(C)OC(CNC(C4CC=CC4)=O)(C2)C3)cccc2nonc12 C1(NC(C=C(C)c2ccco2)=O)CCCN(C(C2CCCC(N(C)C)C2)=O)CC1 c1(C(=O)NC(CNC(C2CC(C#C)(O)C2)=O)C2CCC2)cc(OC)c(F)c(F)c1 C1(NC(C(C)c2ccsc2)=O)COC2(CNC(C3(P(C)(C)=O)CC3)=O)CC1C2 C1(CC)CCN(C(=O)CC2CCCCN2C)C1CCC(=O)NCC(C)(Cl)CC CC1COc2c(NCC3CCC4(C3)CC4(F)F)cnn2C1 C(CC(C)C(=O)N1CCN(C(=O)CN(C(=O)Cc2c(C)n[nH]c2C)C)CC1)OC CC(C)(C)C(CO)C(=O)NC1CC1CNC(=O)CC1NC(=O)NC1=O CCC(C)(F)C(=O)NCCC1(O)CN(C(c2cc(CC(C)C)[nH]n2)=O)C1 N1(C(C2(C#C)CC2)=O)CC2(C(=O)NC(C)CC3CCOCC3)CC1CO2 C1(C(=O)NCCn2cccn2)CCCN(C(=O)CCc2cccs2)CC1 c1(C(=O)OC)cc(SCC=CCNC(=O)C=Cc2ncc(C)[nH]2)n(C)n1 CC(=O)C(C)CC(C)C(=O)N1CCC(C(=O)NC2CCC(O)C2)C1 c1(CNC(C(CN(C)C)NC(C)=O)=O)ccccc1-n1cc(C(C)(C)CO)nn1 C1(CNC(c2c(C)cns2)=O)(NC(=O)CC2CCCC2C)CCCCC1 C1(CC(=O)NC(C)(CO)C2CC2)C2CN(C(C3CC3C3CC3)=O)CC12 c1(CCC)c(C(N2CC(N(C(=O)CCc3ccoc3)C)C2)=O)nnn1CC C=C(Cl)C(C)(C)C(=O)N1CCC1CNC(=O)C(c1cccc(F)c1)(C)O C1(C(=O)NC(c2ccccc2[N+](=O)[O-])CC(=O)OC)NCCC12CCOCC2 C1(O)(C(C)NC(c2cnn(CC(F)F)n2)=O)CCN(C(C2(F)CCOC2)=O)CC1 C1(CNC(CCCCOCC)=O)CN(C(c2cc(C3CC3)n(C)n2)=O)CCC1C n1(CC)nc(C(=O)NC2(C)CC(C(N3CC(C(C)OC)C3)=O)C2)cc1O Cc1nc(N)c(CC(=O)NC2CCCCN(C(=O)CCC3CC3)C2)c(O)n1 C1(NC(c2ccnc(C3CC3)n2)=O)CC12CCN(C(C1CCS1(=O)=O)=O)C2 c1(C(=O)NCC(C)(C2CC2)NC(COC)=O)sc(-c2ccco2)nc1C(F)(F)F C12(C(=O)NCC3(C)CN(Cc4ccc(SC)cc4)C3)CC3CC(C1)CC(C)(C3)C2 N1(C(C2CC(=C)C2)=O)CC(CNC(=O)C(c2ccc(Cl)s2)C)CC12CCC2 Cc1c(C(N(C(C)(C)C)CCNC(c2cnn(C)c2Br)=O)=O)cnn1C1CC1 C1(CNC(C(CC)SC)=O)CC2(CCN(C(=O)Cc3c(C)cnn3C)C2)CO1 CCCCC(CC)C(=O)NC(CN(C(=O)Cc1nn(C)cc1Br)C)CC N1(Cc2cccc(CNC3CC(C)NCC3)c2)CCC2(CCCN(C)C2)C1 C1(C(N2C(CN(C(CNC(=O)OC)=O)C)CCCC2)=O)CCC(C)=C(C)C1 c1(OC)nc(-c2cn(C(C)C(=O)N(C)Cc3ncccc3Cl)nn2)sc1C Cc1cc(=NCC(C)(C)CCCO)[nH]cc1S(=O)(=O)N1CCC(F)(F)C1 C1(NC(CCC=CCC=C)=O)CCCC(N(C)C(C2CCCCCC2)=O)C1 CCN(OC)NC(=O)CC(C)OC1CCCCCC1.C1C(=O)N1 C1(CNC(=O)COCC(F)(F)F)C2CCCC1N(C(c1sccc1C#N)=O)C2 c1(C(=O)NCC2CCCN(C(=O)C(O)C3CC3)CC2)nc2n(c1Br)CCC2 c1(C(C)C)ccc(C(=O)NCC(c2ccccc2)NC(=O)C(C)CF)c(O)c1 C(=O)(C1CCCc2sc(C)nc21)NC1CN(C(c2c(C)sc(Cl)n2)=O)CC(O)C1 c1(CSCC)ccccc1C(=O)NC1CCCC1NC(=O)C(C)C1CCCC1 C1(C(N2CC(C(C)NC(C3CCCC3O)=O)C2)=O)CC12CC(C)(C)C2 C12CN(CC1C(=O)NC)C(=O)c1ccc(cn1)O2.N1(CC)CCC1CNC(C)=O C1(CC)(NC(c2ccon2)=O)CCN(C(=O)C(C)CSC)C1 c1(-n2c(C3CC(C(C)(C)C)C3)nc(C(CCC)C)n2)ccc(F)c(F)c1 n1(CC(=O)NC2CN(C(CCC(=C)Cl)=O)CC2F)cc([N+](=O)[O-])cn1 C1(NC(c2sccc2-n2ccnn2)=O)CCC(NC(C2(C3CCOC3)CC2)=O)C1 CN1CCCC(C(=O)NC2CCC(CNC(=O)C(CC3CC3)CC3CC3)C2)C1 C1(C(=O)NC(CNC(CCN(C)CC)=O)(C)CO)CCc2nc[nH]c2C1 c1(CC(=O)OCC)cnc(SC)[nH]c1=NCCN(C)C(c1cc(C)on1)=O c1(C(=O)NC2(CNC(C(CC)OCC)=O)CC2)ccc(F)c(O)c1F Cc1cnc(C(=O)NC2CC(CNC(C3(O)CCC3)=O)C2(C)C)c(C)c1 c1(CCC(=O)NC2CC(NC(C3N(C(C)C)CCC3)=O)C2)nc2ccccc2[nH]1 c1(CN)cc(OC)ccn1.c1(C(N(C(C)=O)CC)C)cccc(F)c1 C1(C)(C(C)C)CN(C(=O)C(C)OC2CN(C(=O)OC(C)(C)C)C2)CCO1 c1(OC)c(C(N2CCOC(CCNC(=O)C(C)C3CCC3)C2)=O)ccc(Cl)c1C CCC(CC(=O)NCCCCCNC(C1C=CCC1)=O)C(=O)OC(C)(C)C C1(OC)CC2CC(C(c3nnnn3C(C)C)(C)NC3(CN(C)C)CC3)C1C2 c1(C(N2CC(CC(F)F)C2)=O)n[nH]c2c1CN(C(c1ccc3c(c1)CCC3)=O)C2 CCCCC(C(=O)N1CCC(C(N)CC(=O)O)CC1)C(C)C CC(CNC(c1cccc(CO)c1)c1nnnn1CCOC)S(N)(=O)=O CCCC(C)(C)CC(=O)N1CCCC1CNC(=O)C(F)(F)CCc1ccccc1 CC(C(C)(C)NC(=O)C=CI)NC(C1CCCN1C(N)=O)=O C1(NC(=O)NCCn2c(C)ccn2)CN(C(=O)C(C)(C)C)CCO1 C(CC(C(=O)NC(C)CCCO)NC(c1ccc(OC)nn1)=O)=CC O=C(CN=c1cc[nH]cc1)N1CC2(CCN2C(=O)CN2CCC(C(F)(F)F)C2)C1 c1(-c2cc(C)c(C=O)s2)cc2c(cc1O)CCCC2 C1(C(=O)OC(C)(C)C)CCCCN(C(=O)C(=O)NCCC2CCC(C)(C)C2)C1 c1(CNC(C2(COC)CCC2)=O)nocc1C(=O)NCC(CO)N(C)C C(=O)(C(O)CC(N)=O)NCC(C(N1CCC(CCF)CC1)=O)N(C)C C(=O)(C1=CCC(C)CC1)N1CCC(NC(c2cc(C)nnc2)=O)C1 c1(CN2CC3C(NC(C4CC4c4ccsc4)=O)C3C2)cccc2[nH]ncc12 C1(NC(C=CSC)=O)CCN(C(C2CC2c2ccc(OC)c(F)c2)=O)CC1F C(=O)(CC(C)CC(C)C)NCCC(CNC(c1c(C)ccs1)=O)O C1(C(=O)NC(COC)COC)C2CC1N(C(=O)CC1CCCN1C)C2 C12(CNC(C(C=C)c3ccccc3)=O)CC(CN1C(=O)CC1CCC(C)C1)C2 c1(OC)ccc(C(CNC(=O)C(C)(C)C23CC(C2)C3)NC(=O)C(N)=O)cc1 c1(CN2C(C)CC(NC(C3(C(=O)N(C)C)CC3)=O)C2)cc(F)cc(Br)c1F C(CC(=O)Nc1cccc(C)c1C#N)(C(C)(C)C)NC(C#CC1(CC)CC1)=O CC1(C(=O)NC2CC(NC(c3ccc(NC(N)=O)cc3)=O)C(O)C2)CS(=O)(=O)C1 CCC(CC(=O)N1CC2(C)CC1(n1cc(-c3ccc(C#N)cc3C)nn1)C2)C(F)F CC(CC(=O)N1CC(F)(C(=O)NCC(O)(CO)CO)C1)C(F)(F)F c1(C(N2CC(C)N(C(=O)CC3(C)OCCO3)CC2)=O)ccn2nccc2n1 c1(CCC(N2C(CNC(CC(C)SC)=O)CCCC2)=O)c[nH]c2c(C)cccc12 c1(C(=O)NC2CCCN(S(CC)(=O)=O)CC2)cc2ncccc2[nH]1 C=CCCN=C(NCC=C1CCCC1)N1CCC(C(=O)OC)C(F)C1 C(CCC(C)(C)C(=O)N1CCN(C(=O)CCC2CC2(F)F)CC1C)OC CC(C(=O)NC1CCC1C(N1CC(N2CC(F)C2)C1)=O)c1ccco1 c1(C(=O)NC(CC(C)NC(c2nc(C(C)C)oc2)=O)C)cnc(O)nc1O CC1(CNC(C2(CC(F)F)CCC2)=O)CC(NC(=O)Cn2cnc(C(N)=O)n2)C1 C1(N(C(CCC=C)=O)CCO)CCN(C(=O)CC2CC(OCC)C2)CC1 C(=O)(C(O)CCCNC(C1CCOCC1)=O)N1CC(C=C)C1 c1(C(=O)NCCC(=C)CNc2c([N+](=O)[O-])cnn2C)cc2c(s1)CCC(C)C2 C=CCC(C)(C)CNC(C1CCC(CNC(c2ccc(F)cc2)=O)CC1)=O Cn1nnc2c1CCN(C(=O)CCC1CCN(C(=O)COC3CCC3)CC1)C2 C(C)(C)(CC(=O)N1CCC(O)CC1)NC(C=CC(=O)OCC)=O N1(C(CC2(C(=O)OCC)CC2)=O)CCC(NC(=O)Cc2ccsc2Cl)CC1C C1(C)(CNC(c2n(CC)nc(C)c2)=O)CCN(C(c2c(C#N)cnn2C)=O)CC1 C1(F)(CNC(c2cc(CCC)oc2C)=O)COCCN(C(C2(F)CCC2)=O)C1 N1(C(C(C2CC2)OC)=O)CCOCC1CNC(c1ccc(-c2ccccc2)o1)=O c1(C(N(CCCNC(C=CCC)=O)C)=O)cc(C(C)(C)C)ccc1N C1(NC(c2cccc(N)c2)=O)CN(C(=O)Cc2ncncc2Cl)CCC1F N1(C(CC(C(=O)OC)C)=O)CC2=C(C1)CN(C(=O)C1=COCCO1)C2 CN1C(=O)CSC1=CC(=O)NCCC(O)CNC(=O)CCn1cccn1 CC1CN(C(c2ccc(Cl)s2)=O)CCC1N(C(=O)CCc1ccc(F)c(F)c1)C c1(-c2cc(CO)oc2CO)cc(C(=O)NCCOC)c2cc[nH]c2c1 C1(CC(CNC(CC)=O)O)CCCN(C(=O)CCCN2CCCC2)C1 c1(C(=O)NC(C2(O)CN(C(c3cc(CC(C)C)on3)=O)C2)C)cc(Cl)cnc1O C1(C)(CNC(CC2(C)CC2)=O)CN(C(c2nccnc2C(N)=O)=O)CCO1 C(=O)(C(O)C(F)(F)F)NC(CNC(c1c(CC(=O)OC)scc1)=O)(C)CO C(=O)(C(C)(CC)CCC)NCCCCCCN(C(COC(CC)CC)=O)C Cc1cc(Cl)cc(C(N2CCC(N(C(=O)CC(C)CF)CCO)CC2)=O)c1N N1(C(C2(C#C)CC2)=O)CCCC(NC(C2CC(N(C)C)C2)=O)C1 c1(CC2CN(C(=O)NC(c3ccc[nH]3)C)C2)ccccc1 c1(C(=O)OCC)c(C)[nH]c(C)c1S(=O)(=O)NC(CCC1CCCO1)C(N)=O C1(NC(C(C)N(C(C)=O)C)=O)CCCC12CN(C(c1cccc[n+]1[O-])=O)C2 CC(C)(CNC(=O)C(C)(C)C1CCOC1)CC(=O)NOCCC(F)F C1(CNC(c2cn(C(C)(C)C)nn2)=O)CN(C(c2ccsn2)=O)CC1(C)C C1(NC(c2cnc(CC)[nH]2)=O)(CO)CCN(C(=O)Cc2c(C)noc2Cl)C1 C1(C(=O)NC(C2CC(NC(c3c(OC)n(C)nc3)=O)C2)C)CC1C1CCCC1 N1(C(CSC2C(CC(=O)NCC(=O)OC)C2)=O)CC2CC1CC2N1CCNCC1 CC(CC(C)(F)F)C(=O)NCC1CC(NC(c2ccoc2Cl)=O)C(O)C1 CCCCS(=O)(=O)CC(=O)N1CC(NC(=O)Cc2ccc(OCC)cn2)CC1C C(N=c1ccc(C(F)F)n[nH]1)C1CC(OC(C)(C)C)C1 C(=O)(CCCCC(F)(F)F)N(C1CCN(C(c2coc(Cl)n2)=O)C1)C c1(C(=O)NCCCN(CCC)C(C2COCC(C)O2)=O)cc(C)c(CC)o1 c1(C(=O)NC2CN(C(C=C(CC)C)=O)C(C)CC2)oc2ccccc2c(=O)c1C c1(C(N(CC(C)O)CCNC(=O)CC=C(Cl)Cl)=O)ccc2ncsc2c1 C(=O)(CCC1=CCCCC1)N.C1(C2(C)CC2)COC2(C1)CN(C(=O)CC1=CCOCC1)C2 CC1CCN(C(C2CC(CNC(c3ccc([N+](=O)[O-])o3)=O)C2)=O)CCS1 C1(C(C)Nc2cc(N3CCC(CN(C)C)CC3)ncn2)COc2ccccc2O1 c1(C(=O)NCC(CNC(C2C(C)OCCC2)=O)O)cnn2ccccc12 c1(CC)cc(NC(=O)CN2CCCC(C)C2c2ccccc2F)c(C)nn1 C1(C(C)NC(=O)C=CCOc2ccccc2)CCCCN1C(=O)Cc1cnc[nH]1 C1(F)(CNC(C2(CC)CC2(F)F)=O)CCN(C(=O)C(F)F)CC1 CC(C)C(C)CC(=O)N1CCC(c2cn(-c3cccnc3C(=O)O)nn2)C1(C)C C1(C(=O)NCc2ccc(C(=O)NC3CC(CC)C3)s2)COCC(C)O1 c1(CC(=O)NC(CNC(c2c(C)ccs2)=O)(C)CO)ccc2c(c1)NC(=O)C2 N1(C(c2c(C(C)C)onc2)=O)CCC(O)(CCNC(=O)C(C)S(C)(=O)=O)CC1 C(=O)(CC1=CCCCC1)NC(C1CCCN1C(=O)C(C)(C)C1CCCC1)C N1(CC2CCN(C(C(C)C)C3CCCO3)C2)CCOCC1=O.C1C(=O)N1 c1(NC(C)=O)ccc2c(c1)CCN(N1CCN(c3ncc(Cl)cc3F)CC1)C2 C=CCC(C)(C)CCN(C(c1cn(C2(N(S(C)(=O)=O)CC)CC2)nn1)=O)C1CC1 C(CC(F)F)(C(=O)NCCN1CCC(O)C1)NC(c1nc[nH]n1)=O CC#CC1CCN(C(C2(CCNC(=O)C(C)NC(C)(C)CC)CCC2)=O)C1 c1(CC)ncccc1C(=O)N(C(C)C(=O)NC(CN(C)C)CC(C)C)CC C1(NC(C(C)n2ccnc2)=O)CC2CCCC(C1)N2C(c1ccc2c(c1)CC2)=O C(=O)(C(C)C(=O)N1CCC(C)(NC(c2cccnc2C(=O)N(C)C)=O)C1)OC C1(CNC(c2n[nH]c(C)c2C)=O)CCN(C(=O)Cc2cccs2)CC1C C1(C)(NC(=O)NC2C(C=C)OCC2)CN(C(=O)OC(C)(C)C)CC1(F)F c1(Cn2cc(CN(C(C(C)(C)C)=O)O)nn2)cc2c(cc1Cl)NC(=O)C2 Cc1nc2c(o1)CCN(C(C1CN(C(C3(CC4CC4)CCC3)=O)CC13CC3)=O)C2 c1(OC)cccc(NCCC(=O)NC(C)(CNC(=O)CC2CC3CC3C2)CO)c1 Cc1ccc(NC(C2(C)CCCN2C(c2nc(C3CC3)cs2)=O)=O)cc1[N+](=O)[O-] C(=O)(CC1CCc2ccccc21)NC1CC2CN(C(C(C(=C)Cl)(C)C)=O)CC2C1 C(=O)(C(O)CCN(C)C)NCCOC1CN(C(C2N(C)CCC2)=O)C1 c1(C(N2CCC(CNC(C3(CO)CCC3)=O)C2)=O)cnc(O)c2ccccc12 c1(C(N(C(CCNC(Cn2cccc(C)c2=O)=O)C)C)=O)n[nH]c2cccnc12 C(=O)(CN=c1cc[nH]cc1)N1CCN(C(C2C(C)OCCO2)=O)CC12CC2 Cn1cc2cc1C(=O)N2.C1(S(C)(=O)=O)(CNC(c2ccc(Cl)cc2)=O)CC1 CCC(CNC(C1CCCN1N=O)=O)(CC)NC(=O)C=CCOC1CCOCC1 N1(C(c2c(CC)scc2)=O)CC2CC(NC(=O)C(C)C3CCCC3)CC1C2 C(=O)(C(C)(C)N(C)C)NC(C1CCN(C(=O)CCNC(=O)C=CCl)C1)C Cc1cc(C(=O)NCC2(F)CCN(C(c3ccc(O)nc3C)=O)C2)c(O)nn1 N1(C(c2n(C)cc(Br)c2)=O)CC2CC1CN2C(C1CC1(Cl)Cl)=O c1(C(=O)NC2C3(CN(C(CCCC(=C)C)=O)C3)CC2)c(OC)cc(OC)cc1F c1(C(N2C(CC)C(C(=O)NC(C)CCC(C)C)CC2)=O)cc(O)ccc1C c1(C(C(C)NC(=O)NC2CC3(CCO3)C2)OCC)ccccc1F CC1CCN(C(C2CCC(=O)NC2)=O)CC1CNC(c1cc(Cl)nnc1O)=O c1(C(N2CCC(C(=O)OC)C2C)C(=O)NCCC)cc(S(N)(=O)=O)co1 C1(NC(C2C(CCC)C2)=O)C2CC(O)C1N(C(c1ccc(C#N)cc1C)=O)C2 c1(C(=O)NC2(C(=O)NC(C3CCCC3)CO)CC2)ccnc(CO)c1 c1(C(=O)NC2(C)CC(NC(c3cc(C)c(C)[nH]3)=O)C2)cc(O)cc(C#N)c1 C1(C(=O)NC(C2CN(C(c3csnn3)=O)C2)C)CCC2CCCCC2C1 C(=O)(C(C(=O)NCC(C1CC1)N(C(=O)C=Cc1c[nH]nc1C)C)OC)OC Cc1c(Br)c(C(N2CCC(C)(C(N3CC4CC3C(=O)O4)=O)C2)=O)nn1C Cc1nc(Cl)[nH]c(=NC(C)CC(C)NC(c2ccc3n[nH]cc3c2C)=O)c1F C(=O)(C(C)S(C)(=O)=O)NC(CCSC)C(=O)NCC1CCCN1C c1(C(=O)NC2(C(=O)NCCCCNC(N)=O)CC(F)C2)ccn2nccc2c1 C1(NC(C(CC=C)C(C)C)=O)CN(C(=O)C=CC)CC12CCCC2 c1(-n2c(C3CC=CC3)nc(C(C)OCC)n2)ccc(C(N)=O)c(F)c1 c1(C(=O)NCCC2(O)CCN(C(c3c[nH]ccc3=O)=O)C2)ccc2nn[nH]c2c1 O=C1c2ccccc2C(=O)N1NC(=O)c1cccc2c[nH]nc12 C1(C(=O)NCc2ccc(C)nc2)CC12CCN(C(=O)C(C)C1CCCC1)C2 C(=O)(C(CC)(CC)C(=O)OC)NCC1CC(F)(CNC(C2CC(C)(CC)C2)=O)C1 N#Cc1ccc(C(N2CC3CCC(C2)N3C(C2OC3CCC2CC3)=O)=O)c(O)n1 c1(OC)ccc(OC)c(CN(c2cc(CO)on2)Cc2ccco2)n1 C1(NC(c2[nH]cc(C)c2)=O)C2CCN(C(C3CCCN(S(N)(=O)=O)C3)=O)CCC12 c1(Nc2cc(NC(C(C)NC(CC)=O)=O)ccn2)cc(CC)cc(C)c1 C1(CNC(Cc2cc(OC)no2)=O)CN(C(=O)CCCN=[N+]=[N-])C2CCCCC12 C1(NC(CCC2CCN(C(CC3CC(C)(F)C3)=O)C2)=O)(CO)CC2(CCC2)C1 C12(C(=O)NC3C(CNC(COc4cc(C)on4)=O)C3)CCCN(CC1)C2 c1(C(=O)NCCN(C(C23CCCC2CC3)=O)CC)cccc(O)c1C C1(NC(c2c(C)scn2)=O)CC2CCC1CC2NC(C1CCCS1)=O N1(C(CC(C)(C)OC)=O)CCC(C2CCCN(C(C3C(C)C3(F)F)=O)C2)CC1 C(=O)(C(CC(=C)C)NC(C1(C2CC2)CC1)=O)Nc1cccc(CC=C)c1 CC1CN(C(C2(CO)CC2)=O)CC(CCN(C(=O)CC(=O)Nc2nccs2)C)O1 N1(C(C2CCC(CC)O2)=O)CCCC(CCNC(=O)C(C)C23CC(C2)C3)CC1 N1(C(C(=O)N(CC)CC)C)CC2CCCN(C(c3cc(Cl)ccc3F)=O)C2C1 C(C(=O)NC(C)CS(N)(=O)=O)(C(C)(C)O)NC(CCC)=O CCCCCCCCCC(=O)N1CC(CNC(=O)CC2CCCN(C)C2)C(C)C1 c1(C(N(CCCNC(c2scnc2C2CCCC2)=O)CC)=O)nnn2c1CCC2 Cc1cn2cc(C(=O)NCC(C3CC3)NC(=O)C(C)(C)C(N)=O)ccc2n1 Cc1cccc(C)c1C(O)C(N1CCC(C(c2ncc[nH]2)O)CC1)=O C=C(C)CC(C(=O)N(C)CC1CCCN1C(=O)C(O)CCC)OC C1(C(C)(C)C)CCCC(C(C)(C)C)C1.C12(CCCC1)C(=O)NC(CO)CNC2=O N1(C(C(C)OCCC(C)C)=O)CC(NC(=O)C(O)CN(C)C)CC(C)(C)C1 N1(C(c2n(CC)nnc2)=O)CCC(CC)(NC(=O)CCC(C)(F)F)CC1 CC(C)CCCCCC(=O)N1C2CCC1(CNC(C1(CO)CCCCC1)=O)CC2 C1(CNC(C2(C(=O)OC)C(=C)CC2)=O)CCCN(C(=O)C(CC)n2ccnc2)C1 c1(OC)ccc(Cl)cc1CC(=O)NC12CCN(C(=O)Cc3nnc(C)s3)CC1C2 CN1CCC(C)(C(=O)NC2CN(C(=O)C3=NOC(C(C)(C)C)C3)C2)C1=O c1(SC)c(C(N2CCCCC2c2n[nH]cc2I)=O)cccc1[N+](=O)[O-] c1(C(CO)NC(c2ccc(C(C)CN(C)C)cc2)C(C)C)ccc(F)c(F)c1F Cc1nsc2ncc(C(=O)NCCC(O)CNC(c3cccs3)=O)cc12 c1(C(=O)NC2CN(C(CCNC(COC)=O)=O)C(C)(C)C2)ccc(Cl)c(C)c1N C1(CC)CN(C(=O)C=Cc2ccccc2Cl)CCN1C(=O)C(C)NC(C)(C)C N1(C(c2c(COC)cc[nH]2)=O)CCC(C)N(C(=O)C2=CCCCC2C)CC1 C1(C(C)NC(C2(C=C)CC2)=O)CN(C(c2cnn(CCC)c2)=O)CCO1 N1(C(CCCN(C(C2(CC(C)C)CC2)=O)C)=O)CC2(CC(N(C)C)C2)C1 c1(CCCOC(C)=O)ccc(C)cc1.c12cnn(c1)N(CCOC)CCOC2 c1(OC)ccc(C(N2CCC(CNC(C3(C)CC=CC3)=O)C23CC3)=O)c(O)c1 C1(C(N(CCNC(C2C(F)(F)C23CC3)=O)CC)=O)CC(C)(C)OC1(C)C CCCCC(C)C(=O)N1CCCCC1C(C)NC(c1ccc(CC(C)C)nc1)=O c1(C(=O)NC2C(C)CN(C(=O)Cc3ccon3)CC2)ccc2[nH]ccc2n1 C(C(N=[N+]=[N-])C(=O)N1CC(C(=O)NCC2CC3CCC3C2)CC(C)C1)OCC c1(C(=O)OC)cncc(C(N2CCC(O)C2C(N2CCOC(C)C2)=O)=O)c1 N1(C(CCNC(=O)OC)=O)CCOCC1CCNC(c1cn(CC(N)=O)nn1)=O c1(C(N2CCN(C(c3cc4n(c3)CCC4)=O)C3CC23)=O)nc2c(s1)CCC2 C1(NC(CN(C(C)C)C)=O)CCCC(NC(C2CCCN2C)=O)C1 N1(C(C(CCC)OCC)=O)CC2(C1)CN(C(C1COC(C)C1)=O)CCO2 CC(CC(=O)NC1CC(CCNC(c2cc(C(F)(F)F)no2)=O)C1)c1ccco1 C(=O)(C#CC1CCOC1)NCC(C(C)(C)C)NC(c1c(NC)nc(C)cc1)=O C12(C(N3C(CNc4nccc(C(=O)OC)n4)CCC3)=O)CCCN(C1)S(=O)(=O)C2 c1cnn2c1NCCC2.C1(N(C)C)CC2CC1N(CC(=O)N(CCO)CCOC)C2 c1(NC(c2cnccn2)C)cc(N2CCC(c3nn(C)cc3O)CC2)nc(C)n1 CC1CCN(CC(=O)NC2CCC(CCNC(C3CN(C4CCC4)C3)=O)C2)CC1 N1(C(c2n(CC#C)ccc2)=O)CC(N(C)C(c2ncccn2)=O)C(C)(C)C1 CC1=CCSC1C(=O)NC(C(=O)NCC1CCC1CO)C1CCC1 c1(NC(c2cccc(F)c2I)=O)cnc2c(c1)CN(C(c1cccnn1)=O)CC2 C1(NC(C2C(CNC(c3n(CCC)ccc3)=O)CCCC2)=O)CCC(O)C(O)C1 C1(C(N(CC(C)NC(c2csc(NC)n2)=O)CC)=O)C(Cl)(Cl)C12CC2 N1(C(C2CCN(C)CC2)=O)CCOC2(CCN(C(C34CC(C3)C4)=O)CC2)C1 Cc1c(C(=O)NCCNC(=O)C(C)CC(C)C)ccc(Br)c1Cl Cn1cnc2ccc(CN3CC4(C3)SCCC4C(=O)O)cc12 C1(NC(CSC)=O)CCC2(CCCN(C(=O)Cc3csc(S)n3)C2)C1 C1(NC(C(N2CC3C(CN)C3C2)=O)=O)C(OC(F)F)C2CCCC12 c1(C(=O)NCCC(CNC(C(CCOC)C)=O)O)ccc2nnn(O)c2c1 c1(CC)conc1C(=O)N(CC1(CC2CCCC2)CC1)C.c1(C(=O)N)csnc1C CC1CCN(C(C2CC(C)(C)CN2C(=O)CC2CNC(=O)O2)=O)CC1(F)F C(=O)(CCCCCOC1CN(C(=O)NCC(=O)NCCOC)C1)NC C(=O)(CCCC(CC)NC(C1CC(=O)C12CCC2)=O)N(CC(=O)OCC)CC c1(N(C(C(=O)Nc2nc(NC(C)=O)sc2)=O)C(C)C2CC2)cc(C)cc(C)c1 C1(c2n(C)ncc2)OCCCC1C(=O)N(C1CN(C(c2cnsn2)=O)C1)CCO C=C(C)CCC(=O)NCCOCCCN(C(=O)CC1CC1C)C c1(C(=O)NC(CNC(c2cc(C(C)C)[nH]n2)=O)C2CCC2)cc2cccnc2s1 n1(CC)nncc1C(=O)NC1(CO)CN(C(C2CC2c2c[nH]nc2C)=O)C1 N1(C(c2c(C)ccc(C)c2)=O)CCC2(CCC2)C(CNC(C2SCCCS2)=O)C1 C12(C(=O)NC(c3nc(C)on3)(C)C)CC(CO1)N(C(c1cc3occc3[nH]1)=O)C2 Cc1ccccc1COCC(N1CC2CC2(NC(=O)CCC2CCOC2)C1)=O C(CC(F)F)(C(=O)NOCC(C)O)N(C(C12CCC(OC)C1C2)=O)C=C(C)C c1(C(=O)NCC(C)(O)CNC(c2nc(O)[nH]c(=O)n2)=O)cnc2c(c1)CCCO2 C(=O)(C(CNC(=O)CCc1cnn(C)c1)C(C)(C)C)NCCNC(=O)OCC N1(C(CC(CNC(c2c(CC)cccn2)=O)C)=O)CCCC(C)(COC)C1 c1(C(=O)NC2C(CNC(C3N(C)CCC3)=O)CCCC2)cnc2ncnn2c1O N1(C(C)=O)CCOC2CCN(C(=O)Cc3c[nH]c4ccc(C)cc34)CC12.c1ccco1 c1(OC)c(C(c2nnnn2C2CC2)NCC(=C2CCOCC2)F)cccc1Br c1(N2CCC(c3ccc(=N)[nH]c3)CC2)ccnc2c(Br)csc12 N1(C(C2(C#N)CCC2)=O)CCC2(CCC(NC)CC2)C1.C(=O)(C1=C(Cl)CCOC1)N c1(CN=c2scc(OCC)[nH]2)nc2c(s1)CCc1ccccc1-2 C1(SCC)CC(C)CCC1OC1CCCCC1 C#CCC(CC(=O)NCCC(C)(C)OC)NC(=O)C(C)SCC C1(NC(c2c(C)coc2C(C)C)=O)CC2(C(N3CC(C)C3(C)C)=O)COC1C2 C1(CC)CC(C(=O)NCCc2ccns2)CCN1C(=O)C(C)N(C)C(C)=O C(=O)(CN1CCCO1)N(c1ccc(F)cc1)CC=C c1(OCC(=O)Nc2ccc(N)c(F)c2)cc2c[nH]nc2cc1F CCC(C)CC(C(=O)N(CC(C)SC)C)NC(c1cnncc1OC)=O N1(C(C(C)S(C)(=O)=O)=O)CC(C2CCCN(C(=O)CN3C(=O)CCC3=O)C2)C1 C(=O)(C1=CCCCO1)NC1(C(N(CCSC)CC)=O)CC1(C)C c1(CCC(=O)NC(c2ccco2)CNC(=O)CCNC(N)=O)cc(Cl)no1 c1(OCC(=O)NCCCCCNC(C2(C(C)C)CCC2)=O)ccc(F)cn1 C(CC(C)(C)C)(C(=O)N1CCC2CCCC12C(N1CCC(OC)C1C)=O)OC c1(-c2n(C(c3ccncc3)C)ccn2)ccncc1-c1cccc(F)c1 C(C(C)(C)C(=O)NCC1CC(NC(=O)C(c2cccc(O)c2)(C)C)CC1O)OC Oc1ncnc2cc(=NCCCCNc3ccccn3)[nH]cc12 C1(CC)CN(C(c2occ(C)c2C)=O)CCN1C(c1ncc(C)cc1Br)=O CC1(C)CCCC(O)(C(=O)NCC2(NC(=O)CC3(CO)CC3)CCCCC2)CC1 c1(COCC(=O)NCC2N(C(Cc3c(C)ncs3)=O)CC2)ccccc1Cl C1(C)(C(N2CCC(CSC)C2)=O)CCN(C(=O)COC(C)=O)CC1 CC1CN(C(C2CC2F)=O)CC1CNC(=O)C(C)(C)C1CCCC1 Cc1cc2n[nH]cc2cc1-c1cn(C2CCN(C(C3CC(N(C)C)C3)=O)C2)nn1 CC#CCCC(=O)NC(c1ccccc1)C(=O)NCc1cc(C(C)C)[nH]n1 n1(CCC)nnc(C(N2CC3C(CNC(=O)C(=Cc4cnc[nH]4)CC)C3C2)=O)c1N CC(CCC(=O)N1CC(F)(C(N2CC(C)(C(N)=O)C2)=O)C1)N(C)C C1(N(C(C2(OC)CCCC2)=O)C)CN(C(C2CC(NS(C)(=O)=O)C2)=O)CCC1C C1(C(N2C(CC(=O)NC3CC(C#N)C3)CC2)=O)CC(N=[N+]=[N-])C1 C12CC3(C1)CC(C3)N2.c1(C(N)=O)cccc(C(N2CC(O)CC2C2CC2)=O)c1 N1(C(c2cc(CC)[nH]n2)=O)CCCC(CCCC(=O)NCC2(C)CCCCO2)C1 c1(CSC)c(C(N2CCN(C(C3CCO3)=O)CC23CCC3)=O)oc2ccccc12 C1(CC)(CC)CC(NC(c2cccc(N)c2)=O)CN1C(C1CCC2(CCC2)C1)=O c1(C(=O)OC)cnc(NCC2CCC(NC(=O)CNC(=O)C(C)(C)C)C2)c(Cl)c1 c1(CC(=O)NCC(CNC(C(C)N(C)C)=O)O)cc(F)cc2c1OCOC2 Cc1nc(NCCCc2ccc(C)s2)cc(N2CCCC(N(C)C)CC2)n1 N1(C(c2c(CC#N)ccs2)=O)CC2(CNC(c3csnn3)=O)CC(F)(C1)C2 N1(C(CCc2c(C)n(C)nc2)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C(CCO)C1 C(=O)(CC(C(C)OC)NC(C1CC(=C2CC2)C1)=O)NC(CCC)C1CCC1 N1(C(C2N(C)CC(C)(C)C2)=O)CC(NC(C2CCCO2)=O)CC2(CC2)C1 CC(C)(CF)C(=O)NC1CCC(C(=O)NC2CCN(CS(C)(=O)=O)CC2)C1 C1(NC(c2ccc(C)cc2I)c2n(CCSC)nnn2)CCCC(C)(C)C1 CC(N=c1[nH]oc2ccc([N+](=O)[O-])cc12)C(C)n1cncn1 C=CCC(CNC(C1CCOC1C(C)C)=O)C(=O)NCc1nc[nH]n1 C1(CNC(C2C(c3n(C)nnc3)C2)=O)C2CCC(C2)N1C(=O)Cn1cnnc1O c1(CC)ccc(NC(C2CCC=CC2NC(c2c[nH]nc2OC)=O)=O)cc1Cl C12CC3(CCN1C2=O)CC3.C1(C(N(C)CCO)=O)CCN(C)C(=O)C1 C1(NC(C(COC)C)=O)CC2(CCN(C(=O)CCSCc3ccccn3)CC2)C1 N1(C(=O)OCC(C)C)CCC12CCC(F)(F)CC2 N1(C(CC2CC(=O)NC2)=O)CCC(O)(CNC(c2nocc2C(F)(F)F)=O)CC1 C1(CC=C)(C(=O)NCCC(C)CC)CCCN1C(c1cc(C(F)F)[nH]n1)=O N1(C(C2(C)CCCO2)=O)CCC2(CC1)CC2NC(c1csc(Cl)n1)=O c1(CC)cc(F)ccc1C(=O)N(CCCN(C(=O)CC1(N2CCCC2)CC1)C)C C1(NC(C2CCC(C)CC2)=O)CS(=O)(=O)C12CCN(C(C13COC(C1)C3)=O)CC2 C=Cc1ccc(C(=O)NCC2C(C)CCCN2C(=O)COCC)cc1 C1(C(=O)NCC2(CC)CCCCC2)CCCN(C(C2CCC(=O)C2)=O)CC1 c1(C(=O)NCC2C(NC(C(C)=C3CCCC3)=O)COC2)cccc(C)c1O N1(C(c2ccc(C(C)(C)C)s2)=O)CCCCC12CCCCC2 C1(N(C(=O)CC2OCCC2(C)C)C)CC2CCC(C1)N2C(=O)CC1CCCSC1 CCC(O)CC(=O)NCc1nc(C)c(C(=O)NCCC2(C)N=N2)o1 CCCC(C(=O)NC1CC(NC(C2CC3CC2C3)=O)C1)c1cccc(Cl)c1 c1(C(=O)NC(CCCCNC(COC(CC)C)=O)CO)cnc2cccnc2c1 C12(C(N(C)CC3CCN(CC)C3)=O)CC(C)(CN1C(=O)CCNC(=O)CO)C2 c1(OC(C)C(N2CCC(NC(=O)CC(C)(C)C3CC3)C2C)=O)cccc(CO)c1 c1(CN(c2ccccc2)C(c2c(OC)ccs2)=O)ccc(C)nc1 N#Cc1ccccc1C(=O)NCC1CCCCN1C(=O)CC(F)(F)F c1(C(C)(C)CNCC2CCC(NC(c3cccs3)=O)C2)cccc(Cl)c1F O=C(C#CC1(C(F)(F)F)CC1)NCC1C2CCC(C2)N1C(c1csnn1)=O C1(OCC)CC(N=c2ccc(-n3ccnn3)n[nH]2)C1 N1(C(C(C(CC)C)C)=O)CCN(C(=O)Cc2ccn(CC)n2)CC(C)(C)C1 C1(NC(C2(C(C)(F)F)CCC2)=O)CC12CC(NC(=O)C(O)Cn1cncn1)C2 c1(OC)c(C(=O)NCCCCCNC(c2cc(C(C)(C)C)on2)=O)occc1=O n1(CC)cccc(NC(=O)C(n2ccc(C)n2)C)c1=O N1(C(C2N(CC)CC2)=O)CCCC1(C(=O)N(C)Cc1ccsc1)C(C)C C=CC(C)C(=O)N(C(CNC(C1CCS1(=O)=O)=O)C1CC1)C C(=O)(CC(C(F)F)C(C)(C)C)Nc1cc(C)c(NC(C2C(Cl)(Cl)C23CC3)=O)cc1 C1(CC(=O)NCCOC2C(C)OCC2)COCCN1C(C1CC1(F)Cl)=O c1(C(=O)NCCN(C(=O)C(C)CC(C)C)CCC)cnc2[nH]ccnc1-2 C(C(C)C)(C(O)C(=O)NC1CCC(CCNC(=O)CN2C(=O)CCC2=O)C1)OC N1(C(C(CCCC)O)=O)CCCC2(C1)CN(C(=O)COCCO)CCO2 Cc1cc(C)c2c(c1)CCC2NC(C1(C)CCS(=O)(=O)CC1)=O C1(C(N(C(CC)C(=O)OC)C)=O)CN(C(=O)CC2(OC)CCOCC2)CC12CC2 C(=O)(C1CCCc2n[nH]cc21)N1CC(O)(CCNC(c2ccc(C#C)cc2)=O)C1 N1(C(=O)OC(C)(C)C)C(COC(c2ccc(OC=C(F)F)cc2)=O)C2CCCC12 Cc1ccc(C(=O)CCC(=O)NCC(CO)NC(=O)C=Cc2ccccn2)cc1 CC1=NNC(=O)C1CC(=O)NCc1cc(C(=O)NCC2(O)CC2)on1 c1(C(N2C(C(=O)Nc3ncccc3CO)CCC2)=O)cc(Cl)cc([N+](=O)[O-])c1 Cc1cccc(C)c1NC(=O)CCC1CCCN(C(=O)C(CC(C)C)N(C)C)C1 C(N=c1[nH]cnc2cccnc12)C1C2CN(C(=O)C=Cc3cc(Br)cs3)CC21 C1(C(N(CCCC(C)C)C)=O)CCCCCC1NC(C1CCC1C(C)(C)C)=O C1(NC(CC(C)C)=O)CCN(C(=O)OC(C)(C)C)CC1.C12CC(C)N1OC2=O c1(CN2CCC(C(=O)NC3CC4(C3)CC4NC(=O)C3CC3)CC2)cccc(F)c1F C(=O)(C1=CCCN(C(c2ccc3nc[nH]c3c2)=O)C1)NC(C(CC)C)C CN1CCC(CC(=O)NCCCC2(NC(C3CCN(CCF)CC3)=O)CC2)C1=O Cc1nc2ccccc2n1CCCOC(=O)C(O)Cc1c(F)cccc1Cl c1(C(N2CC(F)CC2C)C(=O)NCCCSCC)cc(Cl)c(Cl)s1 N1(CCN(C(c2cscn2)=O)CC)CCN(C(=O)CC2(OC)CC2)CC1 Cc1ccccc1C.N12CCN(CC1)N(N1CCCC1)C(=O)C2.C1(C=O)CS(=O)C1 S(=O)(=O)(c1ccc(F)cc1Cl)Nc1cccc(N2C(=O)NC(COC)C2=O)c1 CCC(C)(C)CC(=O)NCc1cc(C(=O)NC(c2ccccc2)C)n[nH]1 C1(c2nnnn2CC(F)F)(CNC2C(C)(NC(=O)OC)CCC2)CC12CCC2 c1(C(=O)NC(C(C)C)CNC(c2cncc(C(F)F)c2)=O)cc2cccnn2c1 C1(CC(=O)OC)CC(C)(C)CN1Cc1nc(C(=O)OC)c(C)s1 c1(C(=O)Nc2cc(CNC(C(C)SC(C)C)=O)nn2C)ccc(Cl)c(O)c1 C(=O)(CS(=O)(=O)CC)NC(COCC)C(=O)NC1(C2CCCO2)CC1 C(=O)(C(C)C(F)(F)F)N1CCC(C(C)C(=O)NCC(C)C)CC1.C(c1ccoc1)=C c1(OC)cc(C)c(C(N2CCC(C)C(NC(C34CC(F)(C3)C4)=O)C2)=O)c(F)c1 C1(NC(c2n(CCCOC)nnn2)c2conc2C)COCC1(C)C CN1C(=O)N(CC(=O)OCc2cccc(OC(F)F)c2)C2(CCCCC2)C1=O C1(CNC(c2ccc(CO)nc2)=O)CCCCN(C(c2ccccn2)=O)CC1 C(=O)(C(C)C(C)C(C)(C)C)NC(C)CCCNC(c1nc(C(F)(F)F)cs1)=O Cc1cc(=NCCCC(C)NC(C2CCOC3(CCCC3)C2)=O)[nH]c(C(C)C)n1 C1(NC(c2cn(CC)nn2)=O)(COC)CCCN(C(C2CCC(F)CC2)=O)C1 N1(C(=O)OCC)CCc2nc(C)nc(O)c2C1.c12cc3ccccc3nc1N2 C1(CNC(C(C(C)C)C)=O)CCC2CN(C(C3CCOCC3)=O)CCC2C1 C1(C(N(C)CC2N(C(COCCC)=O)CCOC2)=O)Cc2cccc(F)c2O1 Cc1cccc2nc(C(C)OC(c3c[nH]ccc3=O)=O)cn12 C1(NC(C(CCCC)C)=O)CCCCCN(C(c2ncnc3ccsc23)=O)C1 Cc1ccc(C(C)CC(=O)NCCNC(C2CCCN(CC(C)C)C2)=O)cc1 CCCCCC(CC)C(=O)N1CC(N(C)C(C2(N3CCCC3)CCC2)=O)C1 C1(NC(Cc2c(OC)nccc2)=O)CN(C(c2nnccc2C)=O)CCC1F N1(C(COC(C)C)=O)CCN(C)C(CNC(c2ncc(F)cc2F)=O)C1 c1(CN(C(C(=O)NC(C)C)C2CC2(C)Br)C2CC2)cccc(C(F)(F)F)c1 Cc1nsc(C(=O)NC2CC23CC(NC(=O)CCC2CCCCC2)C3)c1N C1(C)(NC(CN(CCOC)C(C2CC(C(C)C)C2)=O)=O)CC(O)C1 c1(NC(C(C)(C)OCC)=O)cccc(NC(=O)CCC2C(=O)ON=C2C)c1 N1(C(=O)Cc2cc[nH]c2)CC2(C(=O)NC3(Cc4ccc(F)cc4)CC3)CCC1CC2 c1(C(N2CC(CN(c3ccnc(Cl)n3)C)C2)=O)cc2n(n1)CC(F)C2 c1(CC(=O)NC2CS(=O)(=O)CC2Nc2cc(C(N)=O)ncn2)cnc2ncccn12 N1(C(CNc2ccc(C)cc2)=O)CCC(C)C(CNC(=O)CC2CC3(CCC3)C2)C1 C1(C)(C(N(CCNC(Cn2c(C)ncc2)=O)C)=O)C2Cc3ccccc3C12 c1(-n2cc(C(=O)NC3C(CNC(c4cocn4)=O)C3)nc2)ccc(Cl)c(Cl)c1 C1(N(C(c2c(C)nsc2)=O)C)CN(C(=O)C(c2ccccc2)C2CC2)CC1(C)C Cc1cc(CC(=O)OC(C)C)n(C)n1.N12CCC(C1)C(=O)N(CCO)C(C)C2=O c1(NC(=O)Cc2ccc(N3CCCC3)cc2)ccc2c(c1)C(O)CC2 c1(C(=O)NC(C(C)NC(CCc2cc(OC)no2)=O)C)ccc2c(n1)CCOC2 CC1CC(NC(=O)C(F)C(F)(F)F)CCN1C(=O)C=Cc1cscn1 c1(C(N2CCNC(c3ccc(Cl)cc3)C2)=O)c(O)cccc1Br C1(C(N2CCC(N(C(c3n(COC)ncc3)=O)CCO)C2)=O)CCC2CC1CO2 c1(OC)c(CC(=O)NCCCN(C(C)C)CC2CC2)cccc1F C1(n2cccn2)(C(=O)NC(CC)CO)CCN(C(c2cc(O)n(C)n2)=O)CC1 Cc1nc(NCc2cn(C)nn2)cc(N2CCC(C)(N(C)C)C2)n1 N1(C(CCCc2onc(CCC)n2)=O)CCCC(N(CC)CC2CCOCC2)C1 N12CCC3(C1)CN(C3)OP(OC(C)C)(=O)CC2=O.c1ccccc1 C(=O)(CCC(=O)N1CCC(CC(C)NC(=O)Cc2cnccc2Cl)CC1)OCC C(=O)(C(C)Cc1cnn(C)c1)NC(C1CN(C(c2cnsn2)=O)C1)C c1(NC(=O)COCC2CC2)ccc(CC2CC(C(=O)Nn3cccn3)C2)cc1 C(=O)(CCCC(O)c1ccccc1)N1CC(N(C(c2nc(COC)sc2)=O)C)C1 C1(CC)CC(C(=O)NCC2(C)CCCN(C(=O)CC(C)(C)O)C2)CCC1=O C1(CNC(C(CC)CC)=O)CC2(CCCC2)CO1.C12(C(=O)O)CC1C2 C12(C(=O)NCC3CN(C(=O)C(O)C4CCC4)C4C3C4)CC3CCC(CC(C3)C1)C2 C1(OC)CCCCC1C(=O)NCCCC(C)(C)NC(=O)C#CC1CC1 CCC(CC(=O)NCC1CC(C)CN(C(c2cc(C(C)C)[nH]n2)=O)C1)C(C)C C1(O)(c2cn(CCCCC)nn2)CCN(C(C23CC(C2)C3)C2CC2)CC1 C(=O)(CC1=CCN(C)CC1)N1CC(CCCCNC(C(C(C)C)F)=O)C1 CC(C)CC(C)C(=O)NC1CCCCC1NC(=O)Cc1cc(Cl)cc(Cl)c1 c1(OCCNCCNC(=O)OC)cnn(C2CNC2)c1 CC(C)C(CC(=O)NCC1CCN1C(c1ccc(CO)s1)=O)c1ccccc1 c1(CN2C3C(C(=O)Nc4ccc(C)c(O)c4C)C(C3)C2)cc2cc(Cl)ccc2[nH]1 C(=O)(C1=NN2CCCN=C2N1)N1CCC(C)C(NC(c2cnsn2)=O)C1 c1(-n2c(NC(C)=O)nc(C3CC3)n2)ccc2c(c1)CCC2.N12CC(CC1(C)C)C2 c1(C(=O)NC2CN(Cc3ccn(C)n3)CC2C#N)cc([N+](=O)[O-])c(F)c(F)c1F c1(C(=O)Nc2c(-c3ccc(CS(C)(=O)=O)cc3)cccn2)ccc(O)c(Cl)c1 c1(C(=O)NCc2ocnc2Cn2cc(CCO)nn2)cnc(SC(F)(F)F)cn1 N1(C(CCc2c(C)ncs2)=O)C2CCC1CN(C(C1COC3(CCC3)C1)=O)C2 CN1CC=C(CCNC(C23CCC(CC2NC(=O)C(O)C2CCCC2)C3)=O)CC1 N1(C(Cn2c(C)ccn2)=O)CCN(C)CC1CNC(c1cnc(O)c(F)c1)=O n1(CC=C)cc(CC(=O)NCC(=O)NCC(=O)NCCCCOC)nn1 C1(NC(CC2C(C)CCO2)=O)CC2CCC(C1)N2C(=O)C(C)(C)C c1(C(N2C(C)CC(CNC(=O)C=CCO)C2)=O)[nH]nc2ncccc12 CCCCCCCC(=O)NC1C2CC1N(C(=O)CCc1ccc(C)cc1)C2 C1(NC(c2c(COC)scc2)=O)CN(C(c2cnc(C)cc2C)=O)CCC1CO CCC(O)C(C)C(=O)NCCOCCNC(C1C(N2CCCCC2=O)C1(C)C)=O N#Cc1ccc(-c2ccc(C3CCOC3=O)cc2)c2ccccc12 CC(C)C(C)C(CNC(=O)CCc1ccc(Cl)s1)N=c1cc(Cl)c(O)n[nH]1 C1(CN(C)C(c2ncccn2)C2CCCC2)CS(=O)(=O)C1(C)C N1(C(c2nc(C)sc2)=O)CCCC(N(C(=O)CC2CCCCC23CC3)C)CC1 C12(CNC(C3CC(C(F)F)C3)=O)CCCC(CN(C(=O)C(O)C(F)(F)F)C1)C2 C1(C(N2CCC(CC(=O)N(CC(C)C(F)(F)F)C)C2)=O)CC1C1(C)COC1 c1(OCC)cccnc1C(N1CC(C)(CNC(=O)CN(c2ccccc2)C)C1)=O C1(F)(C(N2CCC(OCCNC(c3cccc(C(F)(F)F)n3)=O)C2)=O)CC=CCC1 C(=O)(C(CC#CC)NC(=O)CCCCC#N)NCc1cnc(CC)[nH]1 N1(C(C=CC)=O)CC(O)CC1CCC=CCNC(C1CN(S(C)(=O)=O)C1)=O C(C1OCCc2ccccc21)N1CCN(n2c(Cc3c(F)cccc3I)nnn2)CC1 N1(CC2(NC(C=C(C)Cl)=O)CC2)CCN(C(c2[nH]cnc2C)=O)CC1 c1(N2CCCC(C)(CC)C2)ccc(S(=O)(=O)NCC2(C3CC3)CCCC2O)cn1 Cc1nc(C=CC(N2CC=CC2CNC(c2sccc2Cl)=O)=O)[nH]c1C C(=O)(C1=CC(C)(C)C1)N(CC(C(=O)NCc1nc(C)sc1C)C)C CC1=NNC(=O)C1CC(=O)NCC1(NC(C2CC23CC(O)C3)=O)CC1 Cc1cc(C(N2CC(C(N3CCOC(C)(C4CC4)C3)=O)(C(C)C)C2)=O)cc(O)c1 S(=O)(=O)(c1ccc(NCCSC(F)(F)F)c(F)c1)NC1(C)CCC(C)C1 C(=O)(C(C)CC(=O)NC(C(=O)NCc1cnc(C)o1)C(C)(C)C)OC N1(C(c2c(NC)scn2)=O)CCCC(C(=O)NCCNC(C2CC(F)(F)C2)=O)C1 c1(CC(=O)N(CC(CC)NC(=O)CC2CC2C)CC)csc(C2CC2)n1 C=CCC(C(=O)NCCC(C)(C)NC(=O)C(C)Cn1cccn1)C(C)C CC(C)CCC(=O)NCC1(O)CC(CNC(=O)CC2(O)CCOC2)C1 N1(C(C(C)N(C)C)=O)CCC(CNC(=O)CCC(=O)N(C)C)CC1C N1(C(CN(C(C)=O)C)=O)CCC2(CCC(CNC(C34CCCC3C4)=O)OC2)CC1 O=C(C#Cc1ccc(C(F)(F)F)cc1)NC1CCCC(F)(F)C1 c1(CN(C)CC2CCN(C(c3c[nH]nc3-c3ccco3)=O)C2)nnc(S)n1C c1(C(=O)NC2C(NC(COCc3c(C)ncs3)=O)CCCC2)c[nH]c(=N)nc1C C(=O)(C1=CCCCO1)N1CCC(N(C(=O)CC2CCC3CC23)CCOC)CC1 C=CCCCC(=O)NC(C)(CNC(=O)CC1CSCCS1)C1CCC1=C(C)C C(CC1CC1)(CC(=O)NC1CCS(=O)(=O)C1)NC(C1C(=C)C1C(=O)OC)=O C(=O)(CC(C)C(C)(C)C)NC(C(C(=O)N(CC(N(OC)C)=O)C1CC1)(C)C)C C(=O)(C(C)CC(F)(F)F)NC(CC#C)C(=O)N1CC(C(C)(C)O)C1 C1(NC(c2cc(COC)sc2)=O)COC2(CNC(=O)C3=NOC(C)C3)CC1C2 n1(CC=C)cc(C(=O)CCNC(=O)C(COC)NC(=O)OCC)nn1.C(C)(C)(C)O N1(C(CCSC)=O)CC(N=c2[nH]c(Cl)ncc2Br)C(C)(C)C1 N1(C(CCOC)=O)CC2CCN(C(=O)Cn3nc(C)c(C)c3C)CC12 C(=O)(C1=C(Cl)CCCC1)N1C(CNC(C(C)n2cncn2)=O)C(C)(C)CC1 c1(OCOC)cc(F)ccc1CN1CCC(C(=O)Nc2ccc(Br)nc2C)C1 CC1=C(C)CC(C(=O)NCc2ccc(C(=O)NC(C)C3CC3)s2)CC1 N1(C(C(CC2CCC2)OC)=O)CCC=CC1C(N1CCN(C2CC2)CC1)=O N1(C(=O)NC(c2cccc(F)c2)c2cc(CO)on2)CCCC(N2CCCC2)C1 C1(NC(CC=C)=O)CCC12CCN(C(c1cccc(C3COC3)c1)=O)CC2 C1(CNC(C(C(CC)C)O)=O)CN(C(c2cncc(F)c2C)=O)CCC1(C)C c1(C(N(CCNC(COCCCOC)=O)C)=O)ccccc1C1CCC12CCC2 C1(C(=O)NCCCOCCNC(c2n(CCC)nc(C)c2)=O)CCC2C1C2(F)F N1(C(C(COC)C)=O)CC2CC(C(N3CCCC3(C)COC)=O)(C2)C1 C1(NC(C2(C)CCC(=O)CC2)=O)CC2CCC(C1)N2C(=O)C(c1ccccc1)O c1(C(=O)NC2CN(C(Cc3cccc(C)c3)=O)CC2C)ccc(C#N)c(O)c1 CC(O)C(F)(F)C(=O)NCCN(C1CCCCC1)C(C1CC2CCC(C1)O2)=O C1(C(=O)O)CC(=O)N1.N1(C(C(C)C)=O)CCC(c2ccccc2CO)CC1 C(=O)(C(CNC(c1c[nH]nc1Cl)=O)C(C)(C)C)N(CC(C(C)C)C)C C1(NC(c2c(Cl)cn(CCC)n2)=O)CN(C(C2(C3CC3)CC2)=O)CC2(CCC2)C1 Cc1cc(C)nc(SCC(=O)N(CC(O)CNC(C2CCN(C)C(=O)C2)=O)C)n1 Cc1cnccc1C=CC(=O)NCCOC1CCN(C(c2conc2C)=O)C1 C1(CCCC)(C(=O)NC2CC(C)(NC(=O)C(Cc3cnc[nH]3)OC)C2)CCCC1 c1(NC(=O)NCc2nc(C(CC)C)on2)ccc(C)c(C(C)=O)c1 N1(C(Cc2c(C)n(C)cn2)=O)CCN(C(=O)CCCc2ccsc2)C2(CCC2)C1 C(CCCCCCn1cc(CCC(C)O)nn1)NC(c1c(C)n(C)nc1)=O c1(C(N2CC(CC(C)NC(C(C=C)OC)=O)C2)=O)cc(CC)ccc1O N(C(=NCCO)NCC(O)COCCO)N1C(C)COCC1.C1(C)CC1 C12(C(=O)NC3C(NC(CC(CC)CC4CC4)=O)C3)CC3CC(C1)CC(CO)(C3)C2 C12(CNC(C(C)NC(c3cncc(C)n3)=O)=O)CC=CC(C1)OC2 C(C(C(=O)N1CCSC(C)C1)OC)NC(CN(C(C)=O)C)=O c1(CC)sc(-c2nccn2CCC2(O)CCOC2)cc1C c1(NC2C(NC(=O)Nc3cccc(OCC)c3)COC2)cc(OC)cc(OC)c1 N1(C(C2CCC(CC)O2)=O)CCOC2CN(C(=O)CC3CCCC(C)O3)CC12 C1(OC)CC(CCNC(=O)CC(C)C)N(C(c2cncc(-c3cc[nH]n3)c2)=O)C1 C1(C(N2C(CNC(C(C(C)C)(C)C)=O)CCC2)=O)CCC2(CC1)CC2(F)F c1(NC(CC2N(C(C#CC(=O)O)=O)CCC2)=O)nccc2cc[nH]c12 Cc1ccc(CC(=O)NC2CC(C)(NC(C3CC3[N+](=O)[O-])=O)C2)cn1 CN1CCC(NCCC(=O)N(CCCNC(C2C(C)(C)C2(F)F)=O)C)CC1 c1(C(c2nnnn2C)NCCC(C(=O)OC)C)ccc(Cl)c(Cl)c1C C1(CNC(c2cc(C)ncc2C)=O)CN(C(=O)CN2CCCC2C)CC(C)(C)O1 C1(NC(=O)CCC(F)F)CCC2(CCCN(C(c3cnc(Cl)s3)=O)C2)C1 C1(C(=O)OC)CCc2nnn(C3CCC(=O)NC3=O)c2C1 c1(C2N(C(=O)C=Cc3ccsc3)CCC2)ccc(F)cc1Cl N1(C(c2cnc(C)c(N)c2)=O)CC2CN(C(C3CCCCC3C)=O)CC2C1 c1(C(=O)NC2CCC(NC(C3CN(CCC)C(=O)C3)=O)CC2)ccc(F)cc1Cl N1(C(CC(COC)C)=O)CC(C2(Nc3ncccc3C#N)CC2)C1 C=CC1(C(=O)NC(C)C(=O)NCCC)CN(C(=O)CN2CC3CCC2C3)C1 N1(C(C=CC)=O)CC2CC(NC(C3CCC=CCCC3)=O)CC1C2 CC(C)C(C)C(CNC(c1cc(Br)c(C#N)s1)=O)NC(=O)CN1CC(C)C1 C1(CC=C)(C(=O)NCC(CO)NC(=O)COC2CCOC2)CCOC1 C1(C(C)C)C(=O)N(CC)CCS1.c1(C(=O)NC)csc(C(F)(F)Cl)n1 N1(C(C2CC(CCC)C2)=O)CCC2(CCCN2C(=O)CSC(F)(F)F)C1 c1(C(N2CCCN(C(c3c(COC)cccc3)=O)CC2)=O)cnn2cccnc12 N1(C(C)=O)CC(O)CC1C(N1CCCC1CN(C)C(C1C(C)CC1C)=O)=O c1(NCC)cc(Cl)ccc1C(N1CCC(CNC(c2ccon2)=O)CC1)=O C1(O)(CCNC(C(C)SCC)=O)CN(C(c2cc(CO)[nH]n2)=O)C1 C1(NC(C=CC)=O)CCCC12CCN(C(c1ccc(OC(C)C)cc1)=O)C2 CC1CC(CCNC(=O)CCC(C)(C)C)CCN1C(C1(C(=O)N(C)C)CC1)=O C1(C(=O)NCCN(C(c2c(C)nc(C3CC3)s2)=O)C2CC2)CCC2CCCCN12 C(=O)(N=c1ccn(C)[nH]1)N1CCC(O)(Cn2cc(C(C=C)(C)O)nn2)CC1 CCCCCC(C(=O)NCCCC(C)(C)NC(=O)CC1=CCN(C)CC1)C(C)C C1(C(=O)NC(CN2CCN(C(C3CC(SC)C3)=O)CC2)C)CCC2CC1C2(C)C c1(C(=O)NCC2C(NC(C(C)(O)C3CCC3)=O)CC2)cc(N)cnc1Br c1(C(=O)NCC2CCC(NC(CC3CC(CC)C3)=O)C2)nc(O)[nH]c(=O)n1 N1(C(C(C)OC2COC2)=O)CCC2(CNC(=O)CCC3CCCC3)CCCC12 N1(C(C2C(CC)CCC2)=O)C(CNC(=O)CCN2CCOC2=O)CC2COCC12 CC1c2ccccc2CN1C(=O)C(=O)NCC1CC1c1cccc(Br)c1 CCCC(O)CC(=O)N1CC2CC1CN2C(c1cc(COC)ccn1)=O c1(C(=O)NCCN(C(=O)C(F)n2ccnc2)CC)cc(N)ccc1C CC1SCCN(C(=O)C(c2cccs2)C2CNC2)C1c1ccccc1 N1(C(CCCN(C(CC(CC)OC)=O)C)=O)CCC2CC2CC1 Cc1cc(=N)[nH]cc1C(=O)NCC(CO)NC(=O)Cn1nc(O)ccc1=O C1(COC)CN(C(c2cnc(OC)nc2)=O)CCN1C(C1CCOC(C)(C)C1)=O C1(NC(CCC(=O)OCC)=O)CC2CCCC(C1)N2C(=O)Cc1coc(C)n1 c1(CC(=O)NC2CN(C3CN(C(C(C)OC)=O)C3)C(=O)C2)cn2cc(C)sc2n1 c1(CCC(=O)NC2(CC(=O)N(CCC#C)CC)CCC2)cccnc1C c1(COC)cccnc1C(N1CC(NC(c2sccc2C(C)C)=O)C(C)C1)=O N1(Cc2onc(C(C)OCC)n2)CCNC(=O)C1c1ccc(F)cc1 N1(C(C2(CCCC)CCCC2)=O)CCCC(CNC(c2cc[n+]([O-])cc2)=O)CC1 C(=O)(N=c1cc(F)n(C)[nH]1)NC(CN(C)C)CCO C1(CNC(C2(C(=O)NC)CC2)=O)C2CN(C(C3CC(n4ccnc4)C3)=O)CC12 c1(NC(=O)CC2CCCN2Cc2cnco2)cc(Cl)cc2ncoc12 CN1C(=O)OC2CN(C(c3ccc(OCc4ncco4)cc3)=O)CC12 C1(CC(=O)NCCC(C)NC(C2N(CC)CCOC2)=O)CCc2ccccc2C1 c1(C(=O)NC(C)CCNC(C2(c3csc(Br)c3)CC2)=O)cncc(N)n1 Cc1cccc(C(=O)NC2(CO)CN(C(C34CC(CF)(CO3)C4)=O)C2)c1 C1(C(N(C2CC2)CC)=O)CCCN(C(C2(N(C)C)CCC2)=O)CC1.C1CC1(C)C N1(C(c2c(C)nc(C)s2)=O)C(C(=O)NCC2(N(C)C)CC2)CCC12CC2 C1(CNC(C2CC(C)(C)C2)=O)CN(C(c2ccc(O)nc2Cl)=O)C2CCCC2O1 N1(C(C(=O)NC(C)C)=O)CCN(C(=O)C(c2cc(F)c(F)cc2F)=O)CC12CC2 C1(NC(C2(C(C)NC(=O)CSCC#N)CC2)=O)CCC(OC(F)(F)F)C1 CCC(C)CC(C)C(=O)NC1(CN(C)C(c2cccn(C3CCC3)c2=O)=O)CC1 c1(C(=O)OC)cc(NC(C2CCN(C(C3(CO)CC3)=O)C2)=O)cc(C)c1 N1(C(c2c(CC)noc2)=O)CC(C)C(C)(CNC(C2(C)CC(C)(C)C2)=O)C1 Cc1cc(C(=O)NC(C)(C)CCNC(C2(C)CCCC2O)=O)cn(C)c1=O N1(C(C2(OC)CCCC2)=O)CC(NC(=O)COCCN(C)C)C(C)C1 C1(C(=O)NC2CC(C)(C(N3CCC(CC(F)F)C3)=O)C2)CCCCC(=O)N1 O=C(NNc1ncnc2sccc12)c1ccc2ncccn12 CC1(CNC(=O)Cc2cccc(OCC#N)c2)CCCN1C(=O)C1CC1 CCC(CCC(=O)N1CCCCC1CC(=O)NCC1=NOC(C)C1)OC C1(CNC(C(C)Cc2ccccc2)=O)CC(NC(=O)CSc2cccs2)CC1O C1(C(N2CCN(C(c3nc(C)n(C)n3)=O)CC2CCO)=O)CCS(=O)(=O)C1(C)C CC1CC(C(=O)NCC(C)N(C)C(C2(Cl)CC2(C)C)=O)C(C)O1 N1(C(c2c(C)ccc(O)c2)=O)CCC2(CCCC2C(=O)N=c2cc[nH][nH]2)C1 c1(CCC(=O)NCCN(C(=O)C=C2CCSCC2)CCC)cccc(C(F)F)c1 CC1(c2nnc(C3CC3)o2)CCCN(CC2CCC3(CCC3)O2)C1 c1(C(N2CCC(N(C(Cc3c(C)ocn3)=O)CCO)CC2)=O)cn(C)c(=O)n1C CC1C(NC(c2ccccc2)=O)CC2CCC1N2C(c1cc(=O)n(C)cn1)=O C1(C(N2CC(O)(CCNC(=O)CN3CCCNC3=O)C2)=O)CC2(COCCO2)C1 C1(NC(CCN(C(C)=O)C)=O)CC2CCC1N(C(=O)C(C)CC(C)(F)F)C2 c1(CC(C)C)ccc(C(=O)C=O)cc1.C(C)(CCCNC(c1ccn(C)n1)=O)N C(=O)(CCCN=[N+]=[N-])NC(CC(C)C)CNC(=O)C(C)(C)c1cscn1 C1(O)(CNc2cn(CCNC(=O)OC(C)(C)C)nn2)CCSCC1 C=CC(C)CC(=O)NC1CC(N(C(=O)CN2CC3CC3C2)C)C1 C1(C(C)(C)NC(C2CC2C(F)(F)F)=O)CCCN1C(c1ccsc1C(N)=O)=O C(=O)(C(C(CC)CC)OC)NC(CCC)CCCNC(c1cscn1)=O C1(NC(c2ccns2)=O)COC2CN(C(c3ccc(C(F)F)cc3F)=O)CC12 C1(C(N(CCN(C)C)CC)=O)C2CC1N(C(=O)CC1(C)CCC1)C2 c1(C(C(=O)NCC(CC)(C)NC(c2occ(C)c2C)=O)C)cn(C)nc1C c1(C(=O)OC)ccc2c(c1)CCCC2Nc1nnc(C2CC2)n1CCOCCOC C1(C(N(C(C)CCNC(=O)CSCCN(C)C)C2CC2)=O)CCOC2(CCC2)C1 Cc1cc(Cl)c(C(=O)N(CCC(C)NC(=O)Cn2ncccc2=O)C)cn1 c1(C(=O)NCCN(C(=O)Cn2c(-c3ccccc3)nnc2S)C)cc(F)n(C)n1 CN1CCN(Cc2ccc(SC3CC(O)(C(F)F)C3)cc2)CC1 c1(NC)ccc(C(=O)Nc2ccc(C(=O)NC)cc2OC)cc1N.OC c1(C(=O)NC2CCCN(C(=O)CC(O)c3ccccc3)C2)cccn2cnnc12 N#Cc1ccc(=NCCC(=O)OCc2ccc(S(C)=O)cc2)[nH]n1 OC1(C2CCC2)CCN(Cc2cc(Cl)sc2Cl)C1 c1(CC)cncc(C(=O)NCCCC(C)NC(C2CCC(=O)NC2)=O)c1 C(CCN(C)C(c1cnc(O)s1)=O)(C(C)C)NC(c1ccn(CCC)n1)=O N1(C(C2CN(C(C)C)C2)=O)CCN(C(=O)CC2(N(C)C)CC2)CC(O)C1 C1(CNC(c2[nH]cc(C)c2)=O)CC2CCCC2N1C(C1CC2(CCCC2)CO1)=O CCCCC(CNC(=O)CCc1nc(C)c(C)o1)NC(c1cnc(N(C)C)s1)=O Cc1cc(O)ncc1C(=O)NCC1CCCCN1c1cc(O)ncn1 C=CCC(C)(CC)C(=O)NCC1(COC)CCCN1C(=O)Cc1ccc(N)cn1 C(=O)(C1=Cc2ccccc2C1)NC1CCCC(CN=c2c(C)cnc(C)[nH]2)C1 C1(NC(C(C)C2CC2)=O)C2CC1N(C(C1CC(O)(C(F)(F)F)C1)=O)C2 C1(CNC(C(CC)OC)=O)CC(OC)CN1C(c1coc(OC)n1)=O Cc1nc2c(n1C)CN(C(=O)Nc1noc3c1CCCC3)CC2 Cc1cccc(OCC(=O)NCCC2CCN(C(c3csc(C)c3)=O)C2)c1 Nc1ccc2nc(N3CCC(CCNC4CC5C=CC4C5)CC3)sc2c1 c1(OCC)cc(CNCCC2CCCN2C(=O)OCC)ccn1.C(C)(C)(C)O c1(NC(=O)CCC(N)=O)cc(CO)ccc1F.CC1CCN2C1C2=O Nc1cc(Br)cnc1C(=O)NC1CCC1NC(C1CC2CC2C1)=O c1(SC)ncc(CN2CCC(C)(C(=O)NC(C)C3CC3)CC2)c(Cl)n1 C1(NC(CCC)=O)CC2CC(CO)CC2C1.C1(=O)C(O)CN1 C#Cc1cncc(NC(C23CC(CO2)N(C(=O)CCc2cn[nH]c2)C3)=O)c1 c1(N2C(C)CC(NC(=O)COCc3ccccc3)C2)nc(O)c2cnn(C)c2n1 N1(C(C2C(CC)C2)=O)CCCC(CO)(NC(c2cccc(-c3ccncc3)n2)=O)C1 c1(C(=O)NCc2ccc(CNC(C(C)SC)=O)cc2)c[nH]cc(C)c1=O c1(C(N2CC3N(C(C(C)C4CCC4)=O)CC(C3)C2)=O)cc2c(cc1N)OCO2 C(N=c1[nH]c2c(c(=NCCC3CC(O)C3)[nH]1)COCC2)C1(CCO)CCCC1 N1(C(C(CCC)(C)O)=O)CC(NC(c2oc3ccccc3c2Cl)=O)CC2(CC2)C1 C(=O)(C(CC)(CC)CC)NC1(C2OCCN(C(C(C(CC)O)C)=O)C2)CC1 N1(C(C(C)CO)=O)CCN(C(c2cc(Cl)sc2Cl)=O)C(c2ccncc2)C1 N1(C(=O)CSCc2cscn2)CCC(CNC(C2CC3C=CC2O3)=O)CC1 c1(C(=O)NCCN(C(c2ccn(CC)n2)=O)C2CC2)sc(C)nc1C(C)C C(CC(O)C(=O)OC(C)(C)C)NC(=O)C(C1(N(C)C)CCCC1)C1CCCCO1 Cc1ccc(C(=O)NCC2CC23CC3(F)F)c(O)c1Br N12CCC(F)(CC1)C1(N=N1)CNC2=O.C1(OC)CCOC(C(F)(F)F)C1 c1(C(=O)NC(CN(C(C2(OC)CCSC2)=O)C)(C)C)[nH]nc([N+](=O)[O-])c1Cl c1(CC(CNC2C(C)SCC2)O)ccc(C(C)(C)C)cc1 C1(C(=O)NCC(CC)NC(C2(F)CCOCC2)=O)Oc2ccccc2OC1C C1(COCc2nccc(OCCC)c2)CN(C(=O)CC2(OC)CC2)C2(CCC2)C1 CCC(CC)(CO)C(=O)N1CC(F)CC1CC(N1CCC(CC(F)F)C1)=O CC1CN(C(=O)C(F)C(C)(F)F)CCC1CNC(=O)CNC=O c1(N2CC3(C(NC(C=C(C)Cl)=O)CCC3)C2)nc(C)nc2scc(C)c12 C1(NC(C2(C)CCCCO2)=O)CN(C(c2cc(C(N)=O)no2)=O)C2(CCCC2)C1 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1C(C)CN(C(c2c[nH]nc2F)=O)C1 C#Cc1ccc(C(=O)NC(C2CCCC2)CNC(C2CC3CC3C2)=O)c(F)c1 N(C(=NCCc1ccccc1)N1CCSC2(CCCCC2)C1)CCC(C)OC c1(CN2C(CC(=O)NC3CC3F)CCC2)cc(F)c(F)c(Cl)c1F C(=O)(C1=CC2C=CC1C2)NCC1C(C(N(C2CN3CCC2CC3)C)=O)CCO1 N1(C(CNC(CCC)=O)=O)CCCC(Cc2cn(-c3ccc(C)nc3)nn2)C1 N1(CCC(O[Si](C)(C)C(C)(C)C)C)CC(N2CCOCC2)CC(CO)C1 c1(C(N2CCC(NC(CCc3ccc(SC)cc3)=O)C2)=O)ccc(O)cc1F c1(CC(=O)NC(CNC(c2c(CC)nc[nH]2)=O)C)c[nH]c2cccc(OC)c12 CC(C)=C=CC(=O)NCC(C1CC1)NC(c1cnn(CC(C)C)c1)=O C1(C(=O)NC(CC)C(C)(C)C)CN(C(C2C3CCCC23)=O)C2(CCC2)C1 c1(C(=O)NCC(C)CNC(=O)C(C)n2cccn2)cc(C(F)(F)F)ccc1O c1(OC)ccnc(F)c1C(N1CC2CC(NC(=O)C(C)(Cl)Cl)C1C2)=O c1(NC(c2ccc(SCCC)o2)=O)cn(C)c(C(=O)NCCSC)n1 CCC(C)C(=O)C(=O)NCC(C)NC(C1CC(CCO)C1)=O N1(C(C23OCC(C)(C2)C3)=O)CC(NC(=O)CSC(C)(C)C)CC2(CCC2)C1 CC1C(NC(c2cn(CCO)nn2)=O)CC2CCC1N2C(C1CSC1)=O c1(NC(C2CC(CNC(C(=O)N(C)C)=O)C23CCC3)=O)n[nH]c2ccc(F)cc12 N1(C(=O)C2CC2)CCCC(C2CCCN2C(c2coc(C3CCC3)n2)=O)C1 CC(C(C)(C)C(=O)NCC1CNC(=O)C1)NC(=O)CC1CCOC1=O CCCC(CCC)CC(=O)N(C)CC1CCCN1C(=O)Cc1cc[nH]n1 c1(NC(C)=O)cc2ccccc2cc1CNC(=O)C#CC1CCC1 CCCCCC(C)(C)C(=O)NCCN(C(=O)CCC1CCCCN1C)CCC N1(C(c2sc3cc(C)sc3c2)=O)C2CCC1CN(C(=O)C=CC=C(Cl)Cl)CC2 c1(C(=O)NCCN(C)C(c2cn(C(C)(C)C)nn2)=O)cc(N)cc2ccccc12 c1(C(=O)NCC2(O)CN(C(=O)CCC3CCC3)C2)cccc2nncn12 c1(C(N2CCC(OC)(CNC(=O)C=C3CCC3)C2)=O)cccc2nc(O)[nH]c12 C12(COC)CC(NC(C3(C)CCOC3)=O)(CN1C(c1cccnc1N)=O)C2 C1(C(=O)NC2(C)CCN(C(CSCC#C)=O)CC2)CCS(=O)(=O)C(C)C1 C1C(C)C(C)N1.n1(CC(N2CCC2CO)=O)cc(C(N2CCOCC2)(C)C)nn1 Cc1nn(C(C)C)c(Cl)c1C(=O)NCC(C)(O)CNC(=O)C(N1CCCC(C)C1)=O N1(CC)CCOC(C(N2CC(C(N3CCCC(NC(C)=O)C3)=O)C(C)C2)=O)C1 c1(NC(=O)Nc2cn(CC3CC(F)(F)C3)nn2)ccc2c(c1)S(=O)(=O)NC2 c1(OCC)nc(NC2CC(CNC(c3c[nH]cc3CC)=O)C2)ncc1Cl c1(C(=O)NC2CCN(C(c3c(C)nc(C)o3)=O)CC2)ccc(F)c(F)c1N Cc1cccc2cc(C(=O)NCC3CN(C(C4CC(C)(O)C4)=O)C3)cnc12 CCCCCCCC(F)C(=O)NCCC(C)NC(=O)CC12CCCC1C2 N1(C(c2c(C)noc2C(F)F)=O)CCC2(NC(C34COCC(C3)C4)=O)CC2C1 N1(CCCC(=O)Nc2c(F)cc(OC)c(Br)c2)CCn2cccc2C12CCNC2 c1(-n2cnc(C(=O)NCC=CCNC(c3cc(C)c(C)[nH]3)=O)n2)c(F)cccc1F C1(N(C)C)CCCN(C(=O)CC2(C)CCN(C(=O)CC3COCC3(C)C)C2)C1 C1(CC(=O)NCC#CCNC(c2cc(Br)co2)=O)CCCCCC1(F)F C1(NC(C(C)OCC=C)=O)CCC(NC(c2ncc(CC(C)C)s2)=O)CC1 CC1CN(C(C2CC(=O)N(C)C2)=O)CC2(CCN(C(C3(C)COC3)=O)CC2)O1 CC(C)C(C)(CNC(=O)CCC1CCCN(C(C23CCCC2C3)=O)C1)C(C)C c12cccnc1N1CCCC(C1)C2.c1(CNC(C)=O)csc(-c2cnn(C)c2)n1 C1(NC(c2nnc3ccccn23)CC(C)C)CCCC(F)(F)CC1 Cc1cc(F)ccc1NC(=O)C(N1CCC(C2CC2)CC1)c1cc(C(F)F)no1 N#Cc1ccc(NC(c2cncc(-c3cccc(C4CCC4)c3)n2)=O)c(I)c1 CC(C)CC(O)C(C)C(=O)N1C2CCC1C(C(=O)Nc1cncc(CO)c1)C2 c1(C(N2CC3C(CNC(CC(CC)O)=O)(CCC3)C2)=O)cnc2cc(C)ccn12 CN1CCCC1C(=O)NCCC1(C(N2CC(CC(F)F)C2)=O)CCCC1 Cc1cc(S(=O)(=O)NC2CCN(C)C(=O)C2)cc(Br)c1C CCCCC(F)C(=O)NCC1CC2CC2N1C(=O)CN1CCC(F)CC1 CN1CC2(CCN(S(=O)(=O)c3ccc(NCCCF)cc3C#N)C2)OCC1=O c1(C(=O)NC(C(C)NC(C2(C)CCOC2)=O)CO)c(N)cc(F)cc1F c1(CC)oc(C(=O)NC(C2CC2C(N2CCCC2c2ccon2)=O)C)cc1C C(=O)(C(C)C(O)C(C)CC)N1CC=C(CN(C(C2(CCC=C)CC2)=O)C2CC2)CC1 c1(CN2C(C(N3CCCC3c3ccc(Cl)s3)=O)CC(O)C2)ccc2ncnn2c1 N1(C(C(C)C)=O)CCC(NC(=O)Cn2ccc(C(F)F)n2)C(c2ccccc2)C1 c1(SCC(=O)N(C)CC2N(C(C3C(C)C3)=O)CCC2)ccccc1Cl c1(C(=O)NC2CN(C(c3c(CC)n(-c4nccs4)nc3)=O)C2)ccc(F)c(F)c1 C1(C(=O)NC2CCCC(NC(C(CC=C)(C)N(C)C)=O)C2)Cc2cccnc2C1 C(CCCCO)N(C(c1ccnn1C)C(=O)NCCCOC(C)(C)C)C C(C(Cc1nc(-c2cccc(F)c2)nn1-c1cnn(C)c1)C(F)(F)F)OC CCCCCC(F)C(=O)N1CC2CCC(C1)N2C(=O)C(C)(O)COC c1(C(=O)NC2CN(C(c3c(CC)non3)=O)CC2C)cc(C(F)(F)F)ccc1F C(=O)(CC1CCC(=O)c2ccccc21)NCCN(C(C1=CCC(C)CC1)=O)C N1(C(CCOCC#C)=O)CCC(C)(CNC(C2CCOC(C)C2)=O)C1 CC(C)C(C)(Br)C(=O)NC1CN(C(C2CC2c2ccccc2)=O)C1 S(=O)(=O)(c1ccc(C)cc1)NCC(=O)NCC(CC=C)NC(=O)CC(C)C=C N1(C(c2nc(-c3cc(C)c(C)s3)sc2)=O)CC(c2nnc(O)n2C)CC12CCC2 C(C(C(=O)N=c1cc(C)n(CCO)[nH]1)OC)NC(c1c(OC)cncc1)=O c1(C(=O)NC(C(CO)NC(c2c(CC)onc2C)=O)C)ccc2ncsc2c1 c1(CNS(Cc2cc(NC(=O)NCC3=CCSC3)no2)(=O)=O)ccc(F)c(Cl)c1F CCC(C)(O)C(=O)N1CCCC(NC(c2ccccc2Cc2nc[nH]n2)=O)C1 C1(C(=O)NC2CC(CNC(C(C)Cc3ccccc3F)=O)C2)CCC(C)(O)CC1 c1(OC)ncnc(OC)c1C(=O)NC(C)CCCNC(C1COC(C)(C)CO1)=O Cc1cnc(C(=O)NC(C)(C)CN(C(=O)C(C)n2cnnn2)C)cc1C N1(C(C(C)SCC)=O)CC(C2CC2)(C(=O)NOCC)C1 Cc1cccc(C(=O)NC2(C(=O)N(C)CCO)CCN(C)C2)c1F C1(NC(c2nc(C(C)C)sc2)=O)CCN(C(C2CC=CCC2)=O)C(C)C1 c1(C(N2CC(C)C(NCc3c[nH]c4cccnc34)C2)=O)cc(F)cc(F)c1 C1(N(C)C(C2CC2[N+](=O)[O-])=O)CN(C(=O)C(F)=CC2CC2)CC1(C)C C(=O)(C1CCCc2ncnn21)NCC1(O)CCN(C(c2c(F)ccc(C)n2)=O)C1 c1(C(N2CCCCC2CC2CCC2)=O)ccc(F)c(Br)c1 N1(C(COCCC=C)=O)CCC2CCCC12C(=O)Nc1ccc(C)c(C)c1 C1(C(=O)NCCC(=O)N(C2CCCCC2)CC#C)COCCC1NC(=O)C(F)F C1(NC(C2C(C)=CCS2)=O)CC(CN(C)C)N(C(=O)CC2CCNC(=O)C2)C1 c1(C(N2CC(CN(C)C)C(C)(C)C2)C(=O)NC)ccnc2c(Br)cccc12 n1(CCOC)cc(C(=O)NC2CCC2NC(C2(C)CCCO2)=O)nn1 c1(C(N2C(C(=O)NCc3cc(C)no3)C(C)CC2)=O)cccc(=O)n1C c1(C(=O)Nc2c(CC)cc(Cl)cc2)c(N)cc(F)cc1F c1(CC)ccc(C(N2CCC(C)(CNC(=O)CCCCSC)C2)=O)cc1 c1(CN2CC(NC(C(CC)n3ccnc3)=O)C3(C2)CC3)ccc2cc[nH]c2c1 N12CCC(CC(O)C1)C2.c1(-c2cn(Cc3n(C)ncc3)nn2)cn(C)nc1I c1(NC(c2c(OCC)ccc(F)c2)=O)ccc(I)c(C)c1C c1(Cn2c(C3(NCC(CC=C)(C)C)CN4CCC3C4)nnn2)cccc2ccnn12 c1(OC)nccc(C(=O)NCC2(F)CC(CNC(=O)CSC(F)(F)F)C2)c1F C1(C(=O)N(CC(C)N(C)C(c2ncoc2CO)=O)C)(NC(=O)OC)CCCCC1 c1(CNC(C)=O)cccc(NC(C2CCCCS2)=O)c1.N12CCC(C)(C1)C2=O C1(C(N(C2CCN(C(C=CC)=O)CC2)C)=O)CCC2(CCC2)OC1 C(=O)(C(C)(C)C(F)(F)F)NC1C(C(=O)NCc2nccc(C)n2)CC=CC1 C(=O)(NNc1cccc(-n2ccnc2)c1)Nc1ccc(C)cc1C(N)=O c1(C(=O)NC2C(C)CCN(C(=O)CC3CC(F)(F)C3)C2)cc2ccccc2cn1 C(=O)(C1=CS(=O)CCC1)NC(CNC(c1cnc(OC)c(C)c1)=O)CC(F)(F)F c1(NC(C23CC(C(=O)NC4N(C(C)=O)CC(O)C4)(C2)C3)=O)cnc(Cl)c(Br)c1C CC1CC(NC(C2(C(F)F)CCCO2)=O)CN1C(c1ccc(SC(F)F)cc1)=O CS(=O)(=O)CCCC(=O)N1CCC(CNC(C2CC(C(F)(F)F)C2)=O)CC1 c1(C(=O)NC(C)CCNC(C2CC(F)(CO)C2)=O)ccc(N)c(F)n1 c1(C(C)C)cccc(C(=O)N(CCCNC(=O)C(c2ccc(Cl)cn2)(F)F)C)c1 c1(CNC(CN(CC)CC)=O)cccnc1CNC(=O)C=C(C)C C1(Cl)(C(N(CCN(C)C(C2CC(N3CCCCC3)C2)=O)C)=O)CC1(C)C C1(C)(COC)CCN(C(C2CN(C(=O)COC3CCCCC3)CCO2)=O)CC1 c1(C(=O)NCC(CC=C)NC(C2CN(C)C(=O)N2)=O)ccc2c(n1)CCCN2 C1(NC(c2c(CC)ncs2)=O)CCCC(NC(=O)Cc2cccn2C)C1 N1(C(C(=O)NCc2ccc(OCC#C)cc2)=O)CCCC(F)(C(=O)O)C1 CCCC(c1nnnn1CC)(c1ccccc1)NC(c1ccccc1)C1CC1 CC1(C)C2CC1CC(=O)N2.C1(CNC(c2nc(CO)cs2)=O)CCC(CO)CC1 C1(NC(C=C(CCC)C)=O)CC2(CCN(C(=O)C(C)(F)CCCC)CC2)C1 c1(NC(C(CC)Cc2cccc(Br)c2)=O)cn2cc(C)ccc2n1 C1(O)(CCNC(CCC=C(C)C)=O)CCN(C(c2ccnc(O)c2)=O)C1 C(C(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)CC1COC(=O)C1)CC2)=C(C)Cl N1(C(c2ccc(C(CC)=O)cc2)=O)CC(C)C(NC(c2cc(C)cs2)=O)C(C)C1 N1(C(C2CCC(CC)CC2)=O)CC(N(C(=O)CCCOC(C)C)C)C(C)(C)C1 N1(C(c2ccc(N(C)C)o2)=O)C(C(=O)NCc2cc(C(N)=O)no2)CCC12CC2 C(=O)(C(F)(F)C(C)O)NCCN(C(=O)CCCN1C(=O)CNC1=O)CCOC c1(C(=O)NC(CN(C(C(C)N(C)C)=O)C)C)cc2ccc(Br)nc2[nH]1 c1(-n2cc(SCC3(NC(C(C)C)=O)CC3(F)F)nn2)ccccc1OC(C)C c1(CN(C(COCCCC)=O)CCNC(=O)C(=O)NCC)ccc(C2CC2)o1 N1(C(C(=O)NCCSC)c2ccsn2)c2ccccc2C(C)(C)CC1C C1(CN(C(C(C)OCCC=C)=O)C)COCCN1C(=O)Cc1ccsc1 C#Cc1cccc(C(N2CC(CC(C)(C)CNC(=O)CC3CCC3OC)C2)=O)c1 c1(C(C)C)nccn1CCNC(=O)C(CNC(c1cnn(C)n1)=O)N(C)C C1(C2CCCCO2)(C(=O)N=c2cc(CN3CCCC3)o[nH]2)CCCO1 C1(C(N(C(C)C(=O)NCCC)c2nccs2)=O)CC(=O)C1 C1(CNC(=O)CCc2nccs2)CN(C(C2C(F)(F)C23CC3)=O)CC2(CCC2)O1 c1(-c2ccc(C#N)cc2)n[nH]c(=NC(=O)NCCCSC2CC=CCC2)s1 c1(C(C)C)nn(C)cc1C(=O)NCC1CCC1NC(=O)C(c1cnccn1)C C(N=c1[nH]c(CC)nc(Cl)c1C(C)C)C1CCCC(CNC(CC)=O)C1 O=C(C1=NOC2(CCC2)C1)NC1C=CCCC1C(=O)NC1COCC1F c1(C(=O)NC(CC(C)NC(CCS(=O)(=O)NC)=O)C)n[nH]c2c1CN(C)CC2 c1(CC)c(OC)cccc1C(=O)NCC(CC)NC(=O)C(C)Cc1cnn(C)c1 C1(CC(=O)N(CCC(C)NC(c2n(CC)nc(C)c2)=O)C)CCn2cncc2C1 C(=O)(C(C)(CC)C(F)F)NCC(c1cccc(C)c1)NC(c1c(CC)n[nH]c1)=O C(=O)(C(C)(C)C(=O)N1CCCC(CCNC(=O)CCC(N)=O)C1)NC C1(CC(=O)NCCOCCOC)COCCN1C(c1cnccn1)=O Cc1ccc(C(N2CCN(C(C3CC3C3CC3)=O)C(C3CC3)C2)=O)c2c1CCC2 CCCC(C)(CCC)C(=O)NC1CC(CCC(=O)NCC2NC(=O)NC2=O)C1 c1(C(N2CC(N(C)Cc3cccnc3F)C2)=O)cccc(Cl)c1O N1(C(=O)C=CSc2ccccc2)CCCC(CNC(c2ccccn2)=O)C1 c1(C(N2CC(C(=O)NCCc3ccc(C)s3)OCC2)=O)cc(C)c(C)nc1 N1(C(c2occ(C)c2)=O)CCCC(F)(C(=O)N(C2CC3CC3C2)C)C1 c1(NC(COC2CC(NC(C3(C)N(C)CC(OC)C3)=O)C2)=O)cnc(C)c(C)c1C C(=O)(C(C(C)(C)O)NC(=O)C(C)NC(C)=O)NC(c1cnn(C)c1)CC Cc1ccc(C(=O)N(CCC(C)NC(=O)C(C)(C)c2cnco2)C)cc1Br c1(OC)cc(C(=O)NCC2CN(C(C3COCCO3)=O)CCO2)cc(F)c1C#N n1(CC)cnc2c1=C1NC(=NC3CC(C3)N1)N=2.C(CC(O)C(C)C)OC c1(C(CO)NC(N(CC(C)C)Cc2nn[nH]n2)=O)ccc(Br)cc1 C1(C(=O)NCC(CSC)OC)CC=CCN1C(c1ccc(SC)cc1)=O C=C(Cl)CCC(=O)NC1C(C(=O)NCC(C)C(C)O)C1(C)C C(=O)(C(F)(F)C(C)(C)O)NC1CCN(C(CC(C)(C)c2ccccc2)=O)CC1O C(CCC(C)C(=O)NC(Cn1ccnn1)C(=O)NCCCC(C)CO)OC C(=O)(C(F)(F)CC1CCCCC1)NCC1C(NC(C(c2ccncc2Cl)C)=O)C1 N1(C(C=C2CCC(C)CC2)=O)CCC(F)(CNC(C2CC(N(C)C)C2)=O)CC1 C1(CN(CC(=O)OC)CC)Cc2ccccc2CO1.c1(C2C3CCN(C3)C2)ccc(Cl)s1 C=CC(C)C(C)C(=O)NC1CC(NC(=O)CCCNC(c2ccccc2)=O)C1 C(C(C(=O)NCc1ncc(C)[nH]1)NC(=O)CCOC(C)C)SCC Cc1ccc2c(c1)C1(CCN(C(C3CC3C)=O)CC1)CN2C(=O)CC#N CC(C)(C)CC(O)CNC(C1COCCN(C(c2cccnn2)=O)C1)=O c1(OCC)ncc(C(=O)NC2CCC(NC(=O)CN(C)CCO)C2)cc1Br Cc1c(O)ccc(C(=O)NC2(CCCNC(C3CCCNC3=O)=O)CC2)c1C CC(C(=O)NCCn1cc(C(N2CCC2C2CCOCC2)=O)nn1)C(F)F CC1CN(N2CC(C(C)(C)O)C2)CC(C)(C)O1 c1(C(=O)NC2CN(C(C3C(C(=O)OCC)C3)=O)C(C)CC2)cn2cc(C)sc2n1 C1(C(=O)NC2(C)CN(C(CC(CCC)C)=O)C2)(COCC)CCCNS1(=O)=O C1(CNC(CCOCCOC)=O)CCN(C(=O)CSc2cccc[n+]2[O-])C(C)C1 N1(CCC)CCCN(C(=O)CC2(NC(c3ccsc3C#N)=O)CCCCC2)CC1 C(C1CCCC1)=C(C)C(=O)NCCCCCN(C)C(c1sccc1F)=O c1(C(C(N2CC(N(C(c3n[nH]c(C)c3F)=O)C)C2)=O)O)ccc([N+](=O)[O-])cc1 C#CCC(C(=O)N1CCC(CN(C)C(c2cnc(CCCC)s2)=O)CC1)C1CC1 CC1(C)CCN(C(C2CC=CCC2)=O)C(C(=O)NCCC23CC(CO2)C3)C1 C(=O)(C(CCSC)OC(c1ncsc1OC)=O)OC Cc1ccc(C)c(C(C)NC(=O)NCC(n2cncn2)c2cc[nH]n2)c1 C1(NC(Cc2c(C)n[nH]c2C)=O)CN(C(=O)CC2CCNC(=O)C2)CC1N=[N+]=[N-] N1(C(CC(C)OC)=O)CC(NC(C2CCOC(C)(C)C2)=O)CC(C)(C)C1 C(=O)(C(C)(C)CF)NCC(C)NC(c1c[nH]nc1-c1ccco1)=O C12(CNC(C3C(C)(C)C3)=O)CC1CN(C(=O)CCCc1n[nH]c(=N)s1)C2 N1(C(CCCN(c2ccccc2)C)=O)CCN(C(=O)C2=CSCCO2)C2CCC12 c1(OC)ccc(-c2ccc(C3(C(=O)NCc4cnc[nH]4)CCC3)nc2)c(F)c1 c1(C(N(C(C)C(=O)Nc2ccsc2)CC)=O)cnc2n1CCC2 C1(N(C(=O)CSCC(N)=O)C)CCN(C(=O)CC2NC(=O)NC2=O)CC1O C1(CNC(=O)CSc2cccs2)CN(C(c2cccnc2OC(F)F)=O)CCO1 C(=O)(CCC(F)(F)F)N(CCC(NCP(C)(C)=O)=O)CCCC1CC1 N1(C(c2nc(C)[nH]n2)=O)CCc2sccc2C1CNC(C1(Br)CC1)=O CC1=C(C(=O)N2CC(F)(CNC(c3ccc(C(C)(C)C)nc3)=O)C2)CCO1 c1(C(=O)NCC(CN(C)C(c2cc(Cl)nnc2O)=O)O)nc(O)nc(O)c1F C(=O)(CCCC(=O)OC)OC(c1nc(CC)nn1-c1cccc(C)c1)C c1(CC(N2CCC(N(C(C(CSC)OC)=O)C)C2)=O)ccc(F)c(F)c1 c1(OC)ccccc1NC(c1cscc1C(=O)NC1CCC1CSC1CCC1)=O c1(C(N2CCC3(CN(C(=O)CC4CSCCN4)C3)CC2)=O)ccc2ccccc2c1 Cc1nc(SC(F)(F)F)sc1C(N1CC(NC(c2c[nH]c(C#N)c2)=O)CC1C)=O C(C(C)C(C)C(=O)N1CCN(C(=O)CC2CCCS(=O)(=O)C2)C(C)C1)OC CC1CCC(CC(=O)N(C)CCN(C)C(c2occc2Br)=O)C1 C1(CC=C)(NC(c2cc(-c3ccncc3)no2)=O)CN(C(C2CC(F)C2)=O)C1 Cc1ccnc2c(C(=O)NC3C4CC3CN(C(=O)C(C)(C)F)C4)cnn12 N1(C(c2cccc(C#N)c2)=O)C2CCC1CN(Cc1cc3ccccc3[nH]1)C2 C(c1cncc(OC)c1)=CC(=O)N(CCN1CCN(C(C2(C#C)CC2)=O)CC1)C N1(C(C(CSC)OC)=O)C2CC1CN(C(C1(C)CC1C)=O)C2 CC1CN(C(c2c[nH]nc2C(F)F)=O)CC(C)CN1C(=O)C=C(C1CC1)C1CC1 c1(OC)ccc(C(c2nnnn2C2CCC2)NC2CC3CCCC3C2)c(Cl)n1 N1(C(C(CC)(C)CO)=O)CC2CCC1CN2C(=O)CNC(=O)NCc1ccco1 N1(C(c2ccc(OC)o2)=O)CCC2(NC(=O)CN3CCS(=O)CC3)CC2C1 CC(CCC(=O)N(C)CC1CCCN1C(c1ccncn1)=O)N(C)C Cc1ccc(Br)nc1CNC(N1CCCC(C)(F)C1)=O c1(CN2C(C(=O)NC(c3ccncc3)C)CC3(CC3)C2)cc(F)c(Cl)c(Cl)c1 c1(C(=O)NCC(CC)NC(C2(CC)CCCCC2)=O)nccc2[nH]ccc12 N1(C(c2c(CCC)n[nH]c2)=O)CC2(C=C(C(=O)NC(c3scnc3C)C)CO2)C1 CC1Oc2ccccc2N(CCC(=O)NCCc2cccnc2)C1=O C1(NC(CC)=O)CC(NC(C2CC3(C2)CC(C)C3)=O)C12CCC2.C12CN(C1)C2=O c1(OC)cc(Cl)c(C(N2CCCC2CNC(C2CC(=O)NC(=O)N2)=O)=O)cc1Cl C(=O)(C(C)(C)C(=O)N1CCC(O)(CNC(=O)CCNS(C)(=O)=O)CC1)NC N1(CC(=O)NC(C(C)C)C)CC2CCC1C1CN(C(c3ccn(C)n3)=O)CC21 c1(C(c2nnnn2-c2ccccc2)NC2C=CC(C(=O)OC)C2)ccc(F)cn1 c1(OC)ccc(C(=O)NC(C)CC(C)=O)cc1S(=O)(=O)NCC1CCCCOC1 CCCCCCCC(=O)NC(C)CC(C)NC(=O)Cc1cc(F)ccc1F CC(c1cccs1)=CC(=O)NCC1CC1CNC(=O)C(C1CCOCC1)O C(=O)(C(=O)N=c1c(Br)c[nH]cc1Br)ONC(C(C1CCC=CCCC1)(C)C)=O c1(C(=O)OC)cc2cc(Cl)sc2cc1NC(C12CCOC1CC(=O)NC2)=O CC1CN(C(=O)CNC(N)=O)CCCN1C(=O)CN(c1ccc(Cl)cc1)C C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCCCC(NC(CC2CC(OCC)C2)=O)C1 c1(OC)ccc(Cl)cc1NNC(=O)OCOc1ccccc1C N1(CCNC(c2cc(-c3ccn(C)n3)on2)=O)CCC(C)C(COC(C)C)C1 S(=O)(=O)(c1cc(Cl)ccc1OCC(F)F)N1CC(O)CC(C)(C)C1 N12CCN(CC1)c1ccc(cn1)C2=O.C(C(C)(C)N(C=O)C1(C)CC1)OC(C)C CC1CN(C(=O)C=C2CCOCC2)CC(CCNC(c2cc(=O)n(C)cn2)=O)O1 c1(C(=O)NC2CC(NC(C3(C)CNC(=O)C3)=O)C2)cnc2ncccn12 N1(C(C2(C(=O)OCC)CC2)=O)CC(NC(c2cccc(O)n2)=O)C2(CCC2)C1 N1(C(CCCCOCC)=O)CCNC(=O)C1CC.C12C=CC(C1)C(=O)N2 C(=O)(C(C)S(N)(=O)=O)N(C1CCN(C(=O)Cc2cnc(C)o2)CC1)CC C(C1=NOC2CCCC12)NC(C(Cn1cccn1)NC(Cc1c(C)ncs1)=O)=O C1(C(=O)NCC2(CNC(c3cn(CC(N)=O)nn3)=O)CC2)CCC(F)(F)CO1 c1(CCC(N2C(C)CC(NC(c3cc(Cl)cs3)=O)C2)=O)c[nH]c2ccccc12 CC1CC=C(C(=O)N2CCCN(C(c3ccc4sncc4c3)=O)CC2)CC1 c1(C(=O)NC2CCN(C(=O)C=Cc3cc(Br)cs3)C2)ccc2c[nH]nc2n1 N1(C(C(C(C)C)F)=O)CCC2(C1)CN(C(=O)CNC(=O)NC1CCCC1)C2 N1(C(CCCCC#C)=O)CCC2(CC1)CN(C(C1CCC(C)S1)=O)CCO2 C1(NC(CNC(CC)=O)=O)CC(O)CN(C(=O)Cc2csnn2)C1 N1(C(C(CC)Cl)=O)CC(NC(c2sccc2OC)=O)CC(F)(F)C1 N1(C(CC(C)SC)=O)CC2CC(C(=O)NCc3cnccc3N(C)C)C(C2)C1 CC1CCN(C(=O)CN(C)C)CC1CC(=O)N(C1CCC1)C C1(CNC(=O)CC2CCSCC2)CC2(CO1)CN(C(C(CC=CC)C)=O)C2 NS(=O)(=O)C1(C(=O)NCC(CO)NC(=O)COc2ccc(Cl)c(Cl)c2)CCC1 C(CC(C(F)F)NC(C)=O)OC.C(=O)(C(CCC1CC1)OC)OC(C)(C)C C1(=CC(N2CC3C(NC(=O)CS)(C3)C2)=O)C2CC3CC(C2)CC1C3.C1(CO)CCOC1 C1(C(=O)NC2(CCCC(=O)N(C(CC(C)C)C)C)CCC2)COCC1(C)C Cc1ccc(CN2CCC(C)(C(=O)N(CCC#N)C)C2)cc1C C1(C(=O)N(C(C)C(=O)N)C)(C)CC=CC1.N(CP(C)(C)=O)OC c1(C(=O)NCCCCNC(CN(C2CC2)CC)=O)ccc(N2CCCCC2)cc1 c1(CC(=O)Nc2ccc(N3CCN(CCOC)CC3)cc2)ccc([N+](=O)[O-])cc1 C(CN=c1cc(C2CC2)nc(Cl)[nH]1)c1cncc(CO)c1 CC1CC(NC(c2ccn(-c3ccccc3)n2)=O)CN1C(C1CC=CC1)=O C(=O)(C1=CCC2CCC1N2C(=O)CCc1cc(C)[nH]n1)NC1C(OC)CCC1 c1(CC(=O)N(C2CC(C(N(c3ccccc3)CC)=O)C2)C)c(C)cnn1C C(=O)(CCC(C)=O)NCCCN(C(C(C)OCC)=O)C CC(C)(C)CC(=O)N1CC(O)CC1CC(=O)NCC1CCCC(CO)C1 C1(NC(c2cnc(OC)c(F)c2)=O)CCN(C(c2nocc2Cl)=O)CCC1CO C(N=c1ccnc(N2CCC(C3CC3)CC2)[nH]1)c1ccc(CO)o1.N12CCCC1C2 C(c1cccc(F)c1)=CC(N1CCC(O)(CNC(C2(CC(C)C)COC2)=O)C1)=O C12(C(N3CCN(C(C4(COC)CC4)=O)CC3CO)=O)CCCCN1CCC2 c1(OC)[nH]c(=N)nc2sc(C(=O)NC(C)CSC)cc12.C123CC1CN(C2)C3=O Cc1ncc(C(=O)NC2CCC2NC(=O)CSc2nncs2)o1 N1(C(C2CC(F)(F)C2)C(=O)NC2CCOC2)CCC(CCO)CC1 C1(C(N2C(CNC(CCCCOC)=O)CN(C)CC2)=O)CCC2(CC1)CC(O)C2 N1(C(C(=CC2CCCC2)C)=O)CCC2(CC1)CC2C(=O)NC(CCO)C(C)(C)O C(CCc1ccccc1)(C(C)(C)C)Sc1ccc(N(CC(=O)OC)C2CC2)cc1.CO C1(NC(C2CCN(CC)C2)=O)CC12CCN(C(=O)CCCCC(C)C)CC2 CN1N=C(CC(=O)NCC2CC(F)CN2C(C2CC=CCC2)=O)CC1=O c1(CC)ccc(C(c2nnnn2C2COC2)NCCC(O)(CC)C2CC2)c(C)c1 N1(CCC(=O)NCCOCCN(C(C2CC(O)(CC)C2)=O)C)CCP(C)(=O)CC1 C12(NC(CN(C)C(N)=O)=O)CC3CCC(C1C2)N3C(C1CC(S(C)(=O)=O)C1)=O CC(CC(=O)NC1C2CC1N(C(=O)Cc1csc(-c3ccco3)n1)C2)C(F)F C1(C(=O)NC(C)Cc2cccs2)CCCCC1C.c12cnc(nc1)c(=O)[nH]2.C(C)C Cc1cncc(C(=O)NCCC2CCN(C(c3ccon3)=O)C2)c1C c1(C(N2C(C(=O)NC(COCCOC)C)CC2)=O)ccc(C#N)c(C)c1 c1(SCC(=O)N(CC(CC)NC(=O)C(F)C2CCCC2)C)nncn1C1CC1 C12(C(=O)NCC3N(C(COCCOCC)=O)CCC3)CCC(F)C1CC2 C1(CC#C)(C(N2CCC(SC)CC2)=O)CCN(C(=O)C=C2CCCCC2)C1 N1(C(C2C(C)(C)CCN2C(=O)CC2CCCC(=O)N2)=O)CC2(CCCCCC2)C1 C=CC1CN(C(=O)C(F)(F)CN(C)C)CC1NC(=O)CC1CSCCS1 C1(NC(=O)CC2(c3ccccc3)CCCO2)C2CCN(C(C3CC=CCC3)=O)C12 C=CCCC(C(=O)NCCCCOC)NC(=O)CCC1CC1C C(=O)(CCCCCC(C)C)N(C1CN(C(CCc2c(C)nccc2)=O)C1)C C(=O)(C(C)(F)CC)N(C1CCN(C(=O)CCNC(=O)NC)CC1)CCC c1(C(=O)OC)ccc(CC(N2CCCC2CCNC(=O)CN2CCCC2)=O)cc1 c1(OCC(=O)NC2CC(NC(c3cc(C)sn3)=O)C2)ccccc1C(F)F c1(C(=O)NCC2N(C(CCCCOC)=O)CCC2)cc2n(n1)CC(F)C2 N1(C(c2[nH]cc(CC)c2)=O)C2CCC1C(C(N1CCCC1)=O)C2.C12(CC1)C(=O)N2 c1(CN(CC(=O)NCCNC(C23CC2COC3(C)C)=O)C)ccc2c(c1)OCO2 C(=O)(CN=c1[nH]c2c(c(=NCCC3CNC(=O)C3)[nH]1)CCC2)N(CC)CC c1(C(C)(C)C)ncsc1C(=O)NCC1(F)CC(CNC(C2(F)CCOC2)=O)C1 c1(C(=O)NC2CN(CC(C3CC3)OCC)CC2(C)C)ccnc2[nH]cnc12 N1(C(C(C)(C)O)=O)CCCCC(C2CN(C(C3CCC(OC(F)F)CC3)=O)C2)C1 c1(CCOC(C)=O)ccc(Br)c(Cn2ccnc2-c2ccccc2Cl)c1 c1(OC)ccnc(NC2CCN(C3CC(=O)N(C4CCCC4CC4CC4)C3)C2)n1 C(=O)(CCC(F)(F)Cn1cc(COCCO)nn1)N(C)CCN1CCCCC1=O N1(C(=O)CN2CCCC2)CC(C2CC2)(C(N2CCC(CCN(C)C)C2)=O)C1 N1(CC)N=C(C(=O)N2CCC3CN(C(C4CC5CC4CN5C)=O)CC23)CCC1=O Cn1nc2nc1C(=O)NCC1CC(C1)C(=O)C2=O.C(C)(C)(C)OC(=O)NC1CC1 c1(C(=O)NCCNC(C(C(=O)OC)OC)=O)cc(Br)cc2scnc12 c1(C(=O)NCC(CNC(c2c(C)cc(C(F)F)o2)=O)(C)O)cccc(O)c1Cl CCC(C(=O)NC1COCC1NC(C1(n2nccn2)CC1)=O)NC(N)=O C1(C(=O)NCC2C(NC(C3CCC(C(CC)(C)C)CC3)=O)C2)CC2CCCCC12 C1(C)(C(N2CCC(O)(CNC(c3c(CC)cccc3)=O)C2)=O)CCN(C)C1=O c1(C(N2CC(C)C(NC(C3(F)CC(N=[N+]=[N-])C3)=O)C2)=O)cc(O)ccc1F C1(C(=O)NCCC(C)N(C(c2ncc(NC)nc2)=O)C)CCN(C)C(C)C1 S(=O)(=O)(c1ccncc1)N1CC(NC(c2ccnc(F)c2)=O)C(F)C1 C(=O)(C(O)C(C)(C)C)N(CC(C)NC(c1cocc1Br)=O)CC CCCC(CCC)CC(=O)NC1CCOC(CNC(c2cccn(C)c2=O)=O)C1 C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(C2CN(C(C)C)C2)=O)C12CC2 N1(C(c2c(C)onc2)=O)CCC(C(C)(C)C)C(CNC(C2OCCC2(C)C)=O)C1 c1(C(=O)NC(C(C)C)C(C)NC(C2CCCCCC2)=O)cccc(=S)n1O C#CC1(CNC(c2cnc(CNC(=O)C(C)CSC)nc2)=O)CCOCC1 N1(C(CC2CCCC(=O)N2)=O)CC2CC1CN2C(=O)CC=Cc1ccccc1 C1(C(c2cccs2)NC(C(c2ccccc2)NC(CSC)=O)=O)CCS(=O)(=O)C1 N1(C(=O)NC2N(C(CC)=O)CCC2)CCN(C(c2ccc(Cl)o2)=O)CC1CO Cc1nc2ccc(-c3ccc(F)cc3O)cc2o1 N1(C(Cc2ccn(CC)n2)=O)CC(CNC(=O)CC=C(C)C)C(C)C1 n1(CC2N(C(C(C)c3cccs3)=O)CC2)cc(CCN(C)C)nn1 C(=O)(CC(C)C(C)C)N(CC(=O)Nc1cnn(C)c1)CC#C c1(C(N2CC(N(C(c3cc(C)cc(C)c3C)=O)C)C2)=O)cc(F)cc2ccoc12 c1(OC)ccc(C(C)=CC(=O)N(CCNC(c2ccccc2)=O)CC2CC2)cc1 C(=O)(C1=NOCC1)NCC(C1CC1)NC(c1cc(-c2ccn(C)c2)[nH]n1)=O C(C)(CCC(=O)NCC1C=CCN1C(=O)Cn1cncc1C)SC C1(C(=O)NC(C)CNC(c2cnn(CCO)c2)=O)CC2CCC1C21CC1 c1(SCC(=O)NC(c2cn(C3CC3)nn2)CC)ccc(F)cc1 c1(C(=O)NC2(CNC(C=CC)=O)CCCCC2C)cc2c(o1)CCC(C)(C)C2 C1(C(=O)NCC(CC)C#N)CC2(CCC2)CN1C(c1ccc(C#N)c(C)c1)=O CC(CC(N)=O)NC(=O)C(C1CCCCC1)NC(C1CCCCC1)=O C#CCC(CC#C)NC(=O)CC1(NC(C2NC(=O)OC2C)=O)CC1 c1(C(=O)NCC2CCCN(C(c3c(C)cnnc3)=O)C2)cc2ncn(C)c2cn1 Cc1cc([N+](=O)[O-])cnc1NC1CCCC(NC(c2c(F)ccnc2F)=O)C1 CCC(C)(CCC(C)C)C(=O)N1CC(CNC(c2ccnn2C(C)C)=O)C(O)C1 c1(CNC(=NCCCOCC)NC2CC2C)c(C)[nH]c2ccccc12 n1(CC(=O)NC2CCOCC2NC(=O)C2=COCCC2)nnc2c1CCCC2 N1(C(C(CC)N(CC)CC)=O)CCC(C)(NC(c2cnc(N(C)C)cn2)=O)C1 CCC(C(=O)NCC(c1ccccc1)NC(=O)COC)C(C)(C)CC N1(C(c2c(CC)nc(C)cc2)=O)CCCC(N=c2cc(C)c(C#N)c(C)[nH]2)CC1 C#CC1(C(=O)NC(C)CC(C)NC(=O)C(c2cnn(C)c2)=O)CCCC1 C1(C(N2CC(NC(c3cc(OC)no3)=O)C(C)CC2)=O)CC2CCC(C1)C2=O c1(C(=O)NC2C(NC(=O)CCCCc3cnn[nH]3)C2)ncnc(O)c1Br c1(C(N2CCCCCC(F)(F)C2)C(=O)NCCCF)ccc([N+](=O)[O-])c(Cl)c1 C(C)(C)(CC(=O)NCC1(C(=O)NC(c2nc(C)no2)C)CC12CCC2)OC N1(CC2(c3ccc(C(F)(F)F)o3)CCC2)CCCC(N2CCNC2=O)C1 C1(NC(=O)NCc2ncn(C(C)C)n2)CCCCC1Oc1ccncc1 C1(N(C(C(C)OCC=C)=O)C(C2CC2)C2CC2)CC2CCC(C1)N2.C1CC2CCC1C2 CN1CCc2cc(NC(C3CCC(CSc4nc[nH]n4)C3)=O)ccc2C1 c1(OCCOC)ccc(Cl)cc1C(N1CC2CC(NC(C3CCCO3)=O)C1C2)=O C1(CC)CN(C(=O)C(C)Cn2cccn2)CCN1C(=O)CC1CCSCC1 CCCC(CCCO)C(=O)NC1CN(C(=O)CCn2ncn(C)c2=O)CC1(C)C C(=O)(CCCCCCCS(C)(=O)=O)N(CCCNC(C(C(CC)C)O)=O)C CCCCS(=O)(=O)N1CCC(C(=O)NCC2CC(C)N(C(=O)C=CCOC)C2)CC1 Cc1ncc(Cl)cc1C(N1CC(CNC(=O)C(C)C(C)(C)C)CC1(C)C)=O c1(OCC)ccc(C(=O)NC2CN(Cc3cn(-c4ccccc4)nn3)C2)cn1 c1(C(=O)NCc2cc(C(=O)NC3(CC=C)CC3)n[nH]2)ncc(C#N)cc1C C(C(C)(O)C(C)(C)C)NC(C1CCC(NC(CC(C)n2cccc2)=O)C1)=O CC(C)CC(CNC(C12CCC(CC1)C2)=O)NC(C1CCN(C2COC2)C1)=O Cc1c(C(=O)NC2CCCCC2NC(C2CCC2)=O)cc(CC(=O)O)n1C CC(C)(C)CCCCNC(=O)C(C1CN(C(C2CN3CCN2CC3)=O)C1)OC N1(C(CC(=O)NCC#C)=O)CCCC(CNC(=O)CC#N)C1 C(=O)(CC(C(F)(F)F)OC)N1CCCC(F)(CNC(CC(CC)(C)C)=O)C1 c1(C(N(C)CC2C(NC(c3[nH]cc(C)c3)=O)CCC2)=O)cnn2ccnc(N)c12 C1(C)(CNC(C(c2ccc(Cl)cc2)OC)=O)CCN(C(C2OCC2(C)C)=O)CC1 C1(C(=O)NCC2CCCC(CNC(c3nc(C)[nH]n3)=O)C2)C2CCC3C(C2)CC13 c1(C(=O)NCCCCC(C)NC(CSCCOC)=O)nccc2[nH]ccc12 C1(C(=O)NCCOCCNC(C2(C)CC=CCO2)=O)CC2(CCCCO2)C1 n1(CC(=C)C)nnnc1C(c1ccn(C(F)F)n1)NCC(=O)OC(C)(C)C c1(C(=O)NCCC2(NC(COCCCC)=O)CCC2)ccc2nncn2c1 C(=O)(CS(=O)(=O)CCO)N1CC(C)N(C(c2[nH]cnc2C#N)=O)CC1 C(=O)(C(C)(C)CC)NCC(C1CCN(C(=O)CS(N)(=O)=O)CC1)C C1(CC(=O)NCC(C2CCCCC2)NC(C2(CC#N)COC2)=O)CC2CCC1O2 C1(NC(C(n2cc(Cl)cn2)C)=O)CC2CN(C(c3cc(F)cnc3O)=O)CC2C1 C1(CCOC)(NC(C23CCC(C2)OC3)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)C1 N1(C(C(C)NC(CC)(C)C)=O)CCCC1CN(C)C(C1(Br)CC1)=O C(c1ccncc1C)=CC(=O)NC1(C)CCN(C(C(CC)(C)OC)=O)C1 C1(NC(c2cc(C(C)=O)on2)=O)CC2CC(C1)CN(C(=O)C=C1CCOCC1)C2 C(=O)(C(C)C(F)(F)F)NCC(C1CCCCC1)NC(CCCC=C)=O C(=O)(C1=NOC2(CCC2)C1)NCC1(N(C(=O)CC(F)(F)C(F)F)C2CC2)CCCCC1 n1(CC(=O)NC2C(CNC(CNC(=O)OCC=C)=O)C2)nc(O)ccc1=O CCC1=C(C(=O)N2CCC(C(C)NC(C3CCC(CC)O3)=O)CC2)SCCO1 Cc1c(C(=O)NCC(F)CNC(=O)Cc2c[nH]nc2O)c(C(F)(F)F)nn1C C(=O)(CC(F)(F)C(F)(F)F)NCC1CCCN(C(C(CCCC)O)=O)CC1 c1(CNC(CNC(COC)=O)=O)cccc(-n2cc(C(C3CC3)SC)nn2)c1 c1(CC)cccc(Br)c1.c12nnc(s1)NCC(C)(C)NC(=O)NC2 c1(C(=O)NC(C)CCCNC(=O)Cn2ncnn2)ccc2nnc(S)n2c1 c1(OC)c(C(=O)NC2CC3CCC2CN3C(=O)C=CCO)cccc1C#N CCCC(CCC)CC(=O)NC1CC(CCNC(C2C3CCCC23)=O)C1 c1(NC(CCC2N(c3nccc(C#N)n3)CCC2)=O)ccc2ccc(Br)cc2c1 C1(C(=O)OC(C)(C)C)CCC2CN(C(=O)C(=O)Nc3cccc(CC(C)S)c3)CC12 O=C(C#CC1CCOC1)N1CCCN(C(=O)CC=Cc2ccccc2)C(CO)C1 C1(NC(=O)NC(C2CC3CCC2C3)C)CCN(C2CCOCC2)CC1 c1(C(N2C(CNC(C3C(C=C)C3)=O)CC(OC)C2)=O)ccc2c(c1)CCOC2 CN1CCC2CCN(C(=O)C3=C(F)CN(C(C4(C)CCCS4)=O)CC3)C2C1 C1(=CCNC(c2cnon2)=O)CCN(C(c2cccc(CO)n2)=O)CC1 N1(C(C(C(C)C)OC)=O)CC(CNC(c2cnc(CC(C)C)s2)=O)OC(C)(C)C1 N1(C(C(C)=CC)=O)CC2CCC2(C2CC2)C1.n12cc(nn1)CNC(=O)C2 C1(CNC(C(CC#C)O)=O)CC2CCC(C1)N2C(=O)Cc1n[nH]c2c1CCCC2 c1(OC)cc(C(N2CCCC(CF)C2)C(=O)NC2CCCC2)ccc1OC.CCOC C=CC1(CC(=O)NC2CCCN(C(=O)C(C)(C)C(C)C)C2)CCCCC1 CCCC(C)CNC(=O)C(C1CCN(C(=O)CCn2ccc(C)n2)C1)F Cc1cccc(C(N2CCN(C)C(CNC(C3CCCC3O)=O)C2)=O)c1Cl CCCCC(CC)C(=O)N(CCN(C)C(C1OCCN(C)C1=O)=O)C(C)C N1(C(CCNC(C(C)(C)C)=O)=O)CCC2CC1CN2C(=O)CC1CCOC1 CS(=O)(=O)c1cccnc1NCC1CCN(C(C2(C3CCCO3)CCC2)=O)C1 Nc1c(C(N2CCCN(C(=O)C=CC3CCCO3)CC2CO)=O)cc(F)cc1Cl c1(NC(c2c(C)cncc2)C)cnn2c1CCCC2C(=O)OC c1(NC(c2ccccc2)CC=C)nccc(=NCc2cc(O)n[nH]2)[nH]1 C#CC1CCC(CNC(=O)CNC2CC3CCCC3C2)CC1 Cc1cc(C(=O)N(C)CC2CCCN2C(=O)Cn2nnc(=N)[nH]2)nc(C(F)F)n1 N1(C(=O)Cc2cccc([N+](=O)[O-])c2)CCC(N2CC(F)C(F)C2)C2(CC2)C1 N1(C(CC(C)c2ccncc2)=O)CC2CCN(C(=O)C3=NOCC3)CCC2C1 C(=O)(C#CC(C)(C)O)N1CC(O)(CNC(C(C)SC(F)(F)F)=O)C1 c1(NC2CC(F)(CNC(c3cc(CCC)on3)=O)C2)cc(C)c(C#N)c(C)n1 CC(C)(C)C#CC(=O)NCC(CO)NC(=O)CCCCNC(N)=O N1(C(CC)C(N)=O)CCN(C(C23CC2COC3(C)C)=O)CC(O)C1 n1(CC)ncc2c1CC(C(N1CC(CC(C)(C)CNC(=O)C3CC3)C1)=O)CC2.N C1(C(N2C3(C(=O)NCCc4ncn(C)n4)CC(C2)C3)=O)CCC(C#N)CC1 C1(NC(c2c(C)n(C)nn2)=O)C2CC3CN(C(=O)C4=COCCC4)C1C3C2 CC1(C)CC(CN)CN1C(=O)C(N1CCCC1c1ccc(F)cc1F)=O C1(CC(C)NC(N)=O)CCN(C(=O)CCCN(C(c2ccoc2)=O)CCO)CC1 C1(C(=O)NC(C2CCCCN2C)C)CCCC12CCC2 C1(NC(c2ccnc(C)c2C)=O)CC2CN(C(=O)Cn3ncn(C)c3=O)CC2C1 N1(C(CN2CCC(C)C2)=O)CCCCC1CNC(=O)C(N1CCNC1=O)C CCC(C(=O)N1CCC(c2nn[nH]n2)C1)NC(=O)Cc1cnn(C)c1 C(=O)(C1CCCc2[nH]nc(I)c21)NCCNC(C1(COC)CCC1)=O C1(NC(=O)NC(c2ccc(OC)nc2)C(F)(F)F)CCC(=O)N(C)C1 CCCCCC(F)C(=O)NC(C)CCC(N1CC(O)CC1(C)CO)=O C(=O)(CC(C)C(C)(C)NC(C1CC(=C2CC2)C1)=O)N1C(C(=O)NC)C=CC1 C=C=C(C)CC(=O)NC1(C(=O)NCCCc2cnn(C)c2)CSC1 c1(NC(=O)OC)cccc(C(=O)NCC2CC(C)N(C(=O)CCCN(C)C)C2)c1 C1(C)(CCNC(C=CC(C)NC(c2cc[nH]n2)=O)=O)CC1(F)F N1(C(Cc2cc(C)sc2)=O)CCOC(C(N2CC(CO)C(C)(C)C2)=O)CC1 c1(OC)cncc(CCC(N2CCC(C(=O)NCCC3(C)CCCO3)C2C)=O)c1 C1(C(N2CCC(OC)(CNC(=O)Cc3cccs3)CC2)=O)C2CCC3C(C2)CC13 c1(CC)nc(C(N2CCCC2Cn2cc(NC(=O)CCC(C)C)cn2)=O)c(Br)s1 CN1Cc2ccc(C(=O)NCC3CCCCN3C(C3CC4CCC3O4)=O)cc2C1 c1(CC(=O)NC2CN(C(CCc3cc(C)[nH]n3)=O)C2)cnccc1C c1(NC(=O)OC2CCOC2)ccc(CCc2ccc(Cl)cc2)cc1 c1(OC)ncc(NC(=O)CN2CCCC=C(Cl)C2)c(C)n1 C1(CN(C)C(c2c[nH]c(=O)cn2)=O)CCCC(NC(c2cnn(C(F)F)c2)=O)C1 c1(C(N(C(CCNC(C(C=CC)O)=O)C)C)=O)cc2c(C)ccc(F)c2[nH]1 C1(CNC(C(CC)CN(C)C)=O)CCCCN(C(=O)Cc2ncoc2C)CC1 n1(CCCC)c(SCc2cncn2-c2ccncc2)nnc1C(F)CC C(=O)(C1c2c[nH]nc2CN1C(c1nocc1Cl)=O)N1CC2C(C(=O)NC)C2C1 C12CN(CC3CCCC13)C(=O)OC2=O.C1(C(C)C)CC(COC(C)(C)C)CO1 C1(C(=O)NCC(COC)C(C)C)(CC)CCCN(C(=O)Cc2ncn(C)c2C)C1 c1(C(N(C2CCN(C(C(CC)C)=O)CC2)CC(C)C)=O)ccc2cc[nH]c2n1 N1(CC(N2CC(CC(C)NC(=O)CC3CCCC4CC34)C2)=O)CCCNC1=O c1(C(C(=O)OC(C(C)=O)C2CC2)=O)c[nH]c2cnccc12 CN=c1ccc(C(=O)NCC2CCCC2C(=O)Nc2cccc(OC)c2C)c[nH]1 C12(C(N3CC(CNC(=O)C4=CCC4)C3)=O)CC(CO)(C1)OC21CCC1 C1(N(C(C2CCCC2)=O)CC)CCN(C(=O)OC(C)(C)C)C1C1CC1 Cc1nc(-c2cccc(C(F)C(=O)O)c2)sc1Cl N1(C(c2cn(CCO)nn2)=O)CCCc2cc(Cl)cnc21.C12CC(CN1)OC2 N#Cc1ccc(C(N2CCCC2CCNC(C2CCC3(CC3)C2)=O)=O)nc1 Cc1c(Cl)ccc([N+](=O)[O-])c1NC(c1c(CNCc2c[nH]c(Br)c2)nccc1)=O CN1CC2CN(C(C3CCCCCN3C(=O)COC3CC3)=O)CC2(C)C1 c1(C(N(CC(C)(C)NC(C2NC(=O)CC2C(F)(F)F)=O)C)=O)ncnc(O)c1Cl CC(C)CC(O)C(=O)N(C1CCN(C(c2coc(C#N)c2)=O)C1)CCO c1(C(N2CCCC(O)(CO)CC2)C(=O)NCCOC)cc(OC)c(OC)c(Cl)c1 C1(F)(C(N(CC)CC)=O)CCCN(C(=O)CCc2ncccn2)C1 N1(C(c2cnn(CC)n2)=O)CCC2CCC(C1)N2C(=O)CCCCCN=[N+]=[N-] N1(C(CCCNC(C)=O)=O)CC2CCC(CNC(=O)C(C)S(C)(=O)=O)(C2)C1 N1(C(CCc2c(C)nc(C)nc2O)=O)CCC(C2(O)CCN(C(=O)CO)C2)CC1 c1(C(=O)NOCC(N2CCN(C3CC3)C3CC23)=O)cccc2c[nH]nc12 Cc1nn(CC(=O)NCC(C)(O)CNC(C2CCCCO2)=O)c(=O)o1 n1(CC)cnc2c(NCc3cncc(N)c3)nc(N(C)Cc3nc[nH]n3)nc12 CC1CN2CCN1CC2C(=O)NC1CC(NC(=O)C(C)(O)C(F)(F)F)C1 C(=O)(CN=c1cc[nH]cc1)NC1CCC(C)(CNC(c2ccsc2Cl)=O)C1 C(=O)(CC(F)(F)CC)NCC1(C(C)(C)C)CCN(C(C(=O)NCC)=O)C1 c1(COC(C2CN(C)C(=O)N2C(c2cnco2)=O)=O)cc2ccc(F)cc2o1 C(=O)(CCC(=O)N1CC2C(NC(=O)CC3CCC4CC4C3)C2C1)NCC C(CN=c1[nH]c(=NC)[nH]c(=NCC2(CC=C)CC2)[nH]1)OCCC=C Cc1ncc(Cl)cc1CC(N1CC(CNC(c2cccc(CO)n2)=O)CC1C)=O C(=O)(C(F)(F)C(C)O)NC1CC(NC(C2CC(C(=O)OC)C2)=O)CC1O C(N(C)N1CC(C(F)(F)F)CC1C)c1cn(C(C)C)nn1 c1(-c2c(CC)nc(C(=O)O)[nH]2)cccc(C(=O)NN2CC(C)(C#N)C2)c1 c1(C(=O)NCC2C(NC(c3c(C)nc(C)s3)=O)CCCC2)cccc2[nH]ncc12 n1(COC)nc(C(=O)NCC23CC(CO2)N(C(=O)CNC=O)C3)ccc1=O C=CC(CC)CC(=O)N1CCC(CC)(NC(C2CC(CC)=NO2)=O)CC1 CCC(C)(COC)C(=O)NC.C1(NC(C2C(C(=O)OC)OCC2)=O)CCC(CO)CC1 C(=O)(N=c1[nH]nc(CC(F)(F)F)s1)NC(c1cnc(-c2cccc(OC)c2)s1)C Cc1c(NCC2(Br)CC2(F)F)ncnc1NCC1CN(CC(F)F)CCO1 CC1CCOC1CC(=O)NC(C)(CNC(=O)CCN1CCOC1=O)C1CC1 C(=O)(CC(CNC(C1CN(C(N)=O)C1)=O)C1CCC1)NC(c1nn(C)cc1O)C C12CCCCN1C(=O)CCN(CC)C2.C(=O)(C(C)CC)NC(=O)NCC c1(NC(C2C3(CCN(C(c4n(C)ccc4)=O)C3)C2)=O)ccc2sncc2c1 Cc1cc(Cl)c(N(CC(O)COCCCOc2ccccc2)C)cc1[N+](=O)[O-] C12(C(=O)NC34CCCN(C(c5c(C)csc5)=O)CC3C4)CC3CC(C(=O)N1)C2C3 N1(C(C)C)CCCC(C(N2CC3C(NC(c4ccc(O)cc4)=O)C3C2)=O)C1 c1(C(N2CC(C(=O)NCC3CCC3C(=O)O)C2)=O)cccc2c1CCN2 C(c1cccc(OC)c1)=CC(=O)NC(CC)CNC(=O)COCCN(C)C c1(OCC(=O)NC2C3CN(C(C(CCC)(C)O)=O)CC32)nn(C)cc1[N+](=O)[O-] CN1C(=O)OCC1C(N1CC(O)(CCc2cn(CCCCO)nn2)C1)=O c1(C(N(Cc2ccc(C)c(F)c2)Cc2csc(Br)n2)=O)c(C)nc2ncccn12 c1(CN(c2nccc(NCC3(C)CCCO3)n2)C)coc2cc(O)ccc12 C1(NC(c2ccoc2)=O)CC2CN(C(c3cc(Cl)ncc3F)=O)CC2C1 N1(C(c2c(C)nco2)C(=O)NCC2CCCCC2)CCN(CC)C2CCCCC12 c1(-n2cc(C)nn2)ccccc1Cl.C1(C(N(CCNC(=O)C)C2CC2)=O)CCNC1 C1(C(=O)NC(C(C)C)(C)CNC(c2cnc(S)[nH]2)=O)CN2CCN1CC2 C1(NC(CN(C2CC2)CC)=O)CN(C(C2(C)COC2)=O)CCC12CCC2 N1(Cc2ccc(Cn3ncc(C)c3)cc2F)CCOC(C2CCCO2)C1 C1(c2ccc(OC)cc2)CCN(C(=O)CC(C)(F)F)CC1NC(C1CC(=O)N1)=O C(C1CCCCC1)=CC(=O)NC(CNC(C1C(NC(=O)OC(C)(C)C)C1)=O)(C)C N1(C(c2ncc(F)cc2F)=O)CCC2C(C1)CN2C(c1ncn2c1COCC2)=O C1(CN(C(C(C)=CC)=O)C)CN(C(c2ccc(N)c(N)n2)=O)CC12CC2 C1(NC(CC2CCN(C(CCC(=O)NC)=O)CC2)=O)CNC(=O)C12CC2 N1(C(C23C(C)(C)OCC2C3)=O)CCC2(CC1)CN(C(C13CCC(CC1F)C3)=O)C2 C(C)(C)(C(C)CC(=O)NC1CCOCC12CCC2)NC(CCC(=C)Cl)=O Cn1[nH]c(=NC(=O)C2CCCN(S(=O)(=O)c3ccc(Br)s3)C2)c2ccc(Cl)nc12 c1(C(CC)OC)nc(-c2ccc(C)o2)nn1-c1cccc(F)c1 N1(C(C(C)OCCC)=O)CC2COCC2(C(=O)Nc2ccc(C)nc2O)C1 C1(CCNC(CC=CC=C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(F)c1F c1(C(c2c(SC(CN3CC4C(C)(C)C4C3)=O)cccc2)=O)nc(Cl)nc(O)c1F C1(CNC(CN(C(CCC)=O)CC2CC2)=O)CCCC1C(=O)N(C)C.OC N1(C(=O)COc2ccsn2)CCCN(C(C2CC2F)=O)CCC1 N1(C(=O)COc2cncc(Br)c2)CCN(C(=O)CCCF)C(CC2CC2)C1 C1(C(N(CCCN(C)C)CCNC(c2ccsn2)=O)=O)C2Cc3ccccc3C12 N1(C(C2(CCC=C)CC2)=O)CC2CCC1CC2NC(=O)C=C(C)C1CC1 C1(N(C(=O)CC2CC=CCC2)CCC)CCN(C(c2cnc(C)[nH]2)=O)CC1 C(=O)(CC(C(F)(F)F)N(C)C)NCC1(CC)CCCOC1.C1(=O)CCCC(=O)N1 N1(C(C(C=C)NC(C2(C=O)CCCO2)=O)=O)CCC(C)(C(=O)NC)CC1 C1(C(N2C(C(C)NC(COCCC)=O)CCC2)=O)CC(=O)N(C)C1 c1(C(N(CCNC(c2c(CCC)nns2)=O)C2CC2)=O)cc(C)n(CCO)n1 c1(C(N(C2CCCCN(C(CCNC(=O)NC)=O)C2)C)=O)ccc2nccn2c1 C1(NC(c2scc(CNC(CC3(C(=C)F)CCC3)=O)c2)=O)CCCN(C)C1=O c1(OC)cc(C=CC(=O)NC2CC23CC(NC(C2(O)CCC2)=O)C3)ccc1O C(CC(=O)NCC(C)(CO)NC(c1ncc2ccccn12)=O)(C(F)(F)F)OC CCC1=C(C(=O)NC2CN(C(c3cc(C(=O)OC)on3)=O)CCC2C)SCCO1 c1(CC(=O)N(CCNC(CNC(C(CC)CC)=O)=O)CC)cc(F)c(C)cc1F Cn1c(I)cc2c(N3CC4CC3CN4C(c3cc(F)ccc3I)=O)ncnc12 N1(C(C2(CC(C)C)CCC2)=O)CC2(CCN(C(C3(C)COC3)=O)C2)C1 C1(N(C(=O)CSc2ccccn2)C)CN(C(=O)CC2CC(C)(C)C(=O)N2)CC12CC2 N1(C(CC#N)=O)CCC2CN(C(c3ccc4c(O)n[nH]c4c3)=O)CC2C1 N1(C(C)=O)CCCC1C(=O)N(CC(C)O)CCNC(c1cn(CCO)nn1)=O C1(CC(C)NC(C2(F)CCC2)=O)CN(C(=O)COCCSC2CCCC2)C1 N1(C(CCSCC(C)C)=O)CCN(C(C2CC(=O)N(CC3CC3)C2)=O)C2CCC12 C1(C(N(C2CN(C(c3csc(-c4ncccn4)n3)=O)C2)C)=O)(CO)CC(F)(F)C1 C1(C(=O)NCc2nc(CNC(c3nocc3C3CC3)=O)sc2)CN2CCC1C2 C1(Cl)(C(=O)NCC2(CN(C)C(c3ccnc(S)c3)=O)CC2)CC2CCC1O2 CC1CN(Cc2cc(Cl)c(Cl)cc2F)CCCN1C(c1cc2cccnn2n1)=O C1(C(=O)NCCC(O)C2CC2)CCC(C2CC2)C1.C12(CC3(CC3)C1)C(=O)NC2 C(=O)(CC(C(F)F)C(C)(C)C)N(C)CCNC(=O)C(C)(C)NS(C)(=O)=O c1(Cc2cn(C3CCN(C(c4ccn(CCC)n4)=O)C3)nn2)nc(C)cc(C)n1 C(C1CCCCC1)=CC(=O)NC1C=CC(CC(=O)N(C)Cc2nnnn2C)C1 CC1(C)CCN(C(C2CS(=O)C2)=O)CC1C(=O)NC1(c2ccsc2)CC1 C1(NC(C2CC(N(C)C)C2)=O)CC(C(=O)NCC2CC23CC3(F)F)CC1O N1(C(C(CNC(C)=O)(C)C)=O)CC2CCC2(NC(=O)C(O)Cc2cnn(C)c2)C1 N1(C(C=C(CC)C)=O)CCN(C2(C(F)(F)F)CCOC2)CC1 N1(C(CC2(C)CCC2)=O)CCC(n2cc(C(O)C3CC3)nn2)C(O)C1 c1(C(C(=O)NCC(CC=C)NC(=O)COc2ccccc2)C)ccc(F)c(F)c1 N1(C(C(C)OCC)=O)CC(NC(c2ccoc2C2CC2)=O)C(CO)C1 N(C1CCCc2cc(C(=O)O)ccc21)C(Cn1cc(CCNC(=O)NC)nn1)=O c1(CNC2CC(C(N3CCC(N(C)C)CC3)=O)C2)ccc2nonc2c1 N1(C(C(CC)(C)OC)=O)CCCCC12CN(C(=O)C(=O)C(C)(C)C)C2 C1(C(=O)NC(CC)(C)CC)CC12CCN(C(=O)C(C(C)C)C1CCC1)CC2 CC(C#N)CCC(=O)NCCN(C(=O)CCC1CCC(O)CC1)C C(CN=C(NCc1ccoc1)NCC1CCCCO1)N1CCN(CC#C)CC1 C1(OCC)CCCN(C(C2CC(C)N2C(=O)CCC(C)SC)=O)C1 c1(C(N2CC3C(CNC(c4nn(C)c(F)c4)=O)C3C2)=O)noc2c1CCCCC2 CC(C)(C)CC(=O)NCC(=O)NCC1(NC(c2cc(CC3CC3)on2)=O)CC1 c1(C(N2C(CNC(c3c(C)nccn3)=O)CC2)=O)cccc2c1N(C)C(=O)CO2 N1(C(C2C(CNC(c3cn(C(C)C)nn3)=O)CC2)=O)CC=CC12CCCC2 CC1(C(=O)NC2CC(C)(NC(C3CCCN3C3CCCC3)=O)C2)CCC(=O)C1 C(C1c2ccccc2CCN1C(c1c(C)nsc1N)=O)NC(C(CCSC)O)=O N1(CCCC)CCCC(C2CCN(C(=O)C(C(C)C)SC)CC2)CC1 CC1(C)CCc2cc(C(=O)NCC(C)(C)NC(C3CC4CC4C3)=O)ccc2N1 C1(CNC(Cc2ccc(C)s2)=O)CC(C(=O)N(CC(C)C(C)C)C)=NO1 N1(C(C2CC(=O)NC2)=O)CCC(NC(c2scnc2C(F)F)=O)C(O)C1 CC1(C)CC(N=c2ccnc(NCC3(CO)CC4CC4C3)[nH]2)CO1 C(=O)(C1=CC2(CCOCC2)C1)N1C2CCC(C(=O)NCC3CCCCO3)(CC2)C1 C1(CNC(C(=O)NC(C)C)=O)CCCN1C(c1ccc(SCC(F)(F)F)o1)=O Cn1nc(O)cc1C(N1CCCC1(C)CNC(=O)COc1ccc(F)cc1)=O c1(SC)cc(C)ccc1C(N1CC(CNC(=O)C(F)(F)CC2CC2)CCC1C)=O N1(C(Cc2cc(C)[nH]n2)=O)CC(N(C)C(C2CC23CCCC3)=O)C(C)(C)C1 Cc1nc(C(=O)N(C)CCNC(c2ccn3c2CSCC3)=O)c2n1CCCC2 N1(C(C)=O)CCCC1(C)C(=O)NCC1CCCCN1C(C1(N(C)C)CCCC1)=O c1(-c2ccc(CN(C)Cc3c(C)nc(Cl)c(=O)o3)s2)cccc2c[nH]nc12 Cn1cc(C(=O)NC2CCC(NC(c3cnc(C4CC4)nc3)=O)CC2)c(=N)[nH]1 CS(=O)(=O)c1nccc(NC2CCCCC2NC(=O)C2=COCC2)n1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C)C1CNC(c1ccccc1F)=O CC(C)S(=O)(=O)CC(=O)NC(C)(C)CN(C)C(C1CC1Cc1ccccc1)=O N1(C(C2(CC(C)C)CC2)=O)C2CCC1CC(O)(CNC(C1(N(C)C)CC1)=O)C2 C1(NC(C(Cn2cncn2)NC(COCC(C)C)=O)=O)CN(C)CC1(C)C C(=O)(CCS(C)(=O)=O)Nc1c(NC(=O)OCC2(C)CCCC2)scc1 CC1OC2(C)CC1(C(=O)NC1CCCC(NC(=O)CCF)CC1)C2 N1(C(c2cc(COC)on2)=O)CC2CC(NC(=O)C=CSc3ccccc3)C1C2 C(=O)(CCCCC(=O)OCCc1ccc(C(N2C(OC)CN(C)C2=O)=O)cc1)OC N1(C(c2c(C)onc2C2CC2)=O)CC2CCCC2(NC(=O)C(Cl)=CCl)C1 CC1(C)CNC(=O)C1NC(=O)CCOCCN(C(=O)C(C1CCCCC1)F)C1CC1 N1(C(C2C(C#N)C2)=O)Cc2occ(C(=O)NC3CC3C3CCCCC3)c2C1 c1(OC)cc(CNC(=O)C#CCNC(=O)CC(C)C2CC2)ncn1 c1(C(=O)NC(CCN(C(C(C(C)C)SC)=O)C)C)cc2c(nn1)CCC2 Cc1cc(C(N2CCC(O)(CNC(=O)Cn3ccc(C(F)F)n3)C2)=O)cc(C)n1 c1(CC(=O)NC2CCN(C(c3cc(C)[nH]c3)=O)CC2)cccc2nonc12 c1(C(=O)NC2(CO)CN(C(c3c(O)cccc3F)=O)C2)cc(F)c(Br)cc1F Cc1cc(C(=O)NCC2CC3CCC2N3C(=O)C=CC2CCCN2C)nc(C)n1 N1(C(C2(NC(C)=O)CC2)=O)CC(N(C(=O)C#CC(C)C)C)C(F)C1 c1(C(=O)NC2C(NC(CCCn3c(C)ncc3)=O)C2)nc(Br)cnc1N C1(C(=O)NC(C#C)C2CCC2)CC(C)CCN1C(C1CC(=O)NC1=O)=O c1(CCC(=O)NC2C3CN(C(c4ccncc4Cl)=O)CC23)c(F)cccc1F c1(C(N2CCC(O)(CNC(=O)CNc3ccccn3)C2)=O)ccc(O)c(CO)c1 C(=O)(C(C)(C)CO)N(C)CC1N(C(C(C)OCC(C)C)=O)CCC1 CCCC1C(=O)N1C.c1(CC(=O)OC)ccccc1CC#N c1(C(N2CCC3(NC(Cc4scc(C)c4)=O)C(C2)C3)=O)c(S(C)(=O)=O)cnn1C Cc1nc(NCCNC(=O)C=CC(C)(C)C)cc(Cl)n1 c1(C(=O)NC(C2OCCN(C(C3(CCOC)CCC3)=O)C2)C)cc(N)cnc1C Cc1c(F)ccc(Br)c1NC(=O)NC1(C)CC(C)(C)OC1=O C1(CNC(C2(NC(C3C(c4c(C)noc4)C3)=O)CCCC2C)=O)NC(=O)OC1(C)C C(=O)(C(CN(C)C)C(C)C)NCC1N(C(C(COC)N(C)C)=O)CC=C1 C1(=O)CC(CCO)NCCCN1C1CNCCO1.c1(C(C)C2CC2)ccccc1 c1(C(N2CCC(C(C)C(=O)NCC(C)(O)CO)C2)=O)cncc(O)c1 c1(SCC(=O)NC(CNC(CS(CCC)(=O)=O)=O)CO)ccc2c(c1)OCCO2 c1(C(N(CC(=O)NCC2(C)CC=CCC2)CCOC)=O)cccc(O)c1 C=C(C)CCC(C(=O)NC1CC(F)(F)C1)N1CCC(C(=O)OC)(OC)CC1 N1(CCOC)CC(C(N2CC3CC3(NC(=O)C(C)C(C)C)C2)=O)CC1=O C1(C)(CN2CC(CC(=O)OC)C2)COCC(C)(C)O1 C(=O)(C1CCCn2cnnc21)NC1C(Nc2ncc(C(=O)OCC)cn2)CC1 N1(C(C(CC=C)CC)=O)CC(NC(=O)COc2cccc(O)c2)CC12CCCC2 N1(C(C(C(CC)C)O)=O)CCC(F)(F)C(CNC(c2cccc([N+](=O)[O-])c2)=O)C1 c1(N(CC#C)CC2CC2)nnc(Cc2ccccc2OC)n1CCCCCC N1(C(C2OCCN(C(C)C)C2)=O)CCN(C(c2cnc[nH]c2=N)=O)CC1CO C1(C(=O)NC2CC(CNC(c3c(NC)snc3C)=O)C2)CCCCNC1=O c1(CC(=O)NC2CCN(C(c3c(CC)nc(C)[nH]3)=O)CC2)c(F)cccc1Cl C(CCCS(N)(=O)=O)NC(c1cnc(C)cn1)c1n(CCCOC)nnn1 Cc1c(CNC(=O)CCN(C(C2C3CCC(F)C23)=O)C(C)C)nnn1C c1(C(=O)NC(C(C)NC(C2(CC#C)CCCO2)=O)CO)cc(OC)cc[n+]1[O-] C12(CNC(CS(CC)=O)=O)CCC(CN1C(c1ccc(C(C)=O)cc1F)=O)C2 N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2CC2(CNC(c2cnn(C)c2Cl)=O)C1 C(=O)(CS(=O)(=O)NC(=O)CCCNC(C)(C)C)NCC(c1cnn(C)c1)C C(CCCCC(=O)NCC1CCCC1)NC(C1(F)C(C)OCC1)=O N#Cc1ccc(NC(=O)C(C2CCOC2)NC(=O)CCCC2CC2)c(O)c1 CC(C)C(C(=O)N(C1CN(C(C2CC(n3cnnc3)C2)=O)C1)C)n1cccc1 c1(C(=O)NCCCC(C)NC(C(C(CC)O)C)=O)cncc2ccsc12 C1(F)(CNC(CC(C)c2ccco2)=O)CCC(NC(=O)Nc2cccc(Cl)c2)C1 N1(C(C2(CC)CN(C(C3CC(=O)NC(C)C3)=O)C2)=O)CCC2CCC(O)C1C2 C1(NC(c2ccc(-c3ccco3)nc2)c2n(CC)nnn2)CC2(COCCO2)C1 c1(C(=O)Nc2ccc(-c3ccc(C(F)(F)F)cc3)cn2)cncnc1Br N1(C(C(c2ccc(N)cn2)C)=O)CCCC12CCN(C(=O)C(F)(F)C1CC1)C2 C1(NC(CN(C)C(=O)C2CC2)=O)CC2CC1N(C(C1(C)CC=CC1)=O)C2 C1(CNC(c2c(OC)nsc2)=O)CN(C)CCN1C(c1cnn(C(C)C)c1N)=O c1(CC(N2CCC(CNC(c3ncc(Cl)cc3Cl)=O)C2)=O)ncn2c1CCCC2 c1(CCNC(CC2N(C(CN(C(C)=O)C)=O)CC2)=O)ccc(C)cc1 c1(C(=O)NCC2C=CC(NC(CC3CC(C)C3)=O)C2)cc(C(F)F)n(C)n1 c1(N2CCN(C3C(c4ccccc4)(O)CO3)CC2)ncnc2sccc12 C(c1cnc(O)nc1O)=CC(=O)NCC(C)NC(c1ccc(Br)c(O)n1)=O N1(C(C(C)Oc2ccccc2Cl)=O)CCN(C(=O)CCn2cccn2)C(C)C1 n1(CC#C)c(C)cc(C(=O)NCC(C)(C)NC(C2CCC(C)O2)=O)c1C c1(NCCN(C(=O)Cn2cnnn2)C)c(F)cccc1[N+](=O)[O-] CC(CCC(=O)NOCc1ccccc1F)NC(C1CCN(C)C1)=O N1(C(c2scc(C)c2C)=O)CC2CCOC2(CNC(c2cc(N)ccn2)=O)C1 CC1CCN(C(c2ccc(C(F)(F)CF)cc2)=O)CC1CNC(C1OCCO1)=O C1(CNC(C2CC(=C)C2)=O)CN(c2nc(C)ncc2F)CCC12CCC2 CCC(C)C(C)C(=O)NCCC(=O)NCc1ccc[n+]([O-])c1 C1(C)(NC(N(CCCN(C)C)C)=O)CC(C)(C)C1 C1(C(N2CCC(N(C(=O)C(=Cc3cccs3)C)CCC)C2)=O)CCCC(F)(F)C1 C(=O)(CCCC(=O)NC(C)C)N(CC(CN(C(c1c(C)cc(F)s1)=O)C)O)C C(C)(C)(CC(=O)NC1CCOC1=O)N(C)C(C1CC1Cl)=O N1(C(CCOC(C)C)=O)CCC(C)C(NC(C2CCS(=O)(=O)C2)=O)C1 C(C)(N=c1nc2c(cnn2C)c(NCCc2sncc2Br)[nH]1)c1c(C)noc1C N1(C(Cc2c(C)cc(Cl)nc2)=O)CCC(NC(=O)CC2=CCCC2)C(F)(F)CC1 N1(CCNC(C2CC(OC)C2)=O)CCN(C(=O)CN2CCCC2CO)CC1 N1(C(CCC2CCC(C)O2)=O)CC2CC(NC(=O)C=Cc3cnn(C)c3)C2C1 C(=O)(C(F)(F)C(O)C1CC1)NCC1CN(C(C(N2CCSCC2)C)=O)C1 CCC(CC)CN=c1[nH]c(=NC2CCCSC2)c2cc(OC)ccc2[nH]1 N1(C(c2cc(C)sc2C)=O)CCC(NC(C2C3COCC23)=O)C2(CCC2)C1 C1(NC(C(c2ccc(C)o2)C)=O)CN(C(c2ccnn2C2CC2)=O)CC12CCC2 c1(NC(C(CC)N(C(=O)CC2CC3CC3C2)C)=O)ccc2nncn2c1 C12(NC(CCCC)=O)COC(CNC(=O)Cn3cc(Cl)c(C)n3)(C1)C2 C1(CNC(C(COC)(C)O)=O)CC(C)CCN1C(c1cnn(CCO)c1)=O c1(NCC(C2CCOC2)OC(C)C)ccc(C(=O)C(C)(C)C)cc1 C12(C(=O)NCC3N(C(c4ncc(OC)nc4)=O)CCCC3)CCN(C1)S(=O)(=O)C2 c1(NC(=O)CCNC(CO)CC(O)c2ccccc2)cc(F)cc(F)c1 c1(C(=O)OC)cc(C(=O)NCC2CCC2NC(c2ccc(F)cc2)=O)ccn1 C12(C(N(CCCC)CCO)=O)CCCC1CCN2C(C1CC2(C1)CC2(F)F)=O CC(C)C(C(C)NC(=O)CSCC(N)=O)NC(=O)CN1CCCCC1 c1(C(=O)NC2C(C)CN(C(C3CC=CC(O)C3)=O)C2)cncc2n[nH]cc12 c1(C(=O)NC2CCN(C(C(C)(C)NC(C)=O)=O)C2)cc(F)c([N+](=O)[O-])c(F)c1 S(=O)(=O)(c1c[nH]ccc1=NC1CCC1C)C(=O)NCCOCCC=C CC1=C(C(=O)N2CC(C)(C)CC2C(=O)NCC2(CO)CC23CCC3)CCC1 c1(C(=O)NCCCN(C(C(C)(C)C(F)F)=O)C2CC2)cc2c(s1)CCCCC2 C1(C(N2CCC(C)(NC(c3cc(C#N)no3)=O)C2)=O)CCCC2CCCN12 c1(N(CCN)CC)ccccc1F.c1(=O)c(=O)n1C.CCCCN(CCCO)C C1(F)(CNC(=O)COC2CCOC2)COCCN(C(c2ncccc2CO)=O)C1 c1(C(N(CCC)CCNC(=O)CCC2CCCC2)=O)noc(CC)c1C N1(C(C2(C)CCNC2=O)=O)C2CCC1(CNC(c1cnncc1O)=O)CC2 C1(NC(c2c(C)n(-c3ccc(F)cc3)nn2)=O)CCC(O)C(O)CC1 C(=O)(C1=NOC(C)(C)C1)NC(CCNC(CN(C)CCc1ccccc1)=O)(C)C c1(C(N2CC(C3(NC(C(C)NC(N)=O)=O)CC3)C2)=O)ccc(F)c(S(N)(=O)=O)c1 CCC(CC)(CN=c1cc[nH]cc1S(=O)(=O)NC(C)CCO)c1ccccc1 CCC(CC(=O)N1CCN(C(C)CNC(=O)C(C)(O)COC)CC1)CC(C)C C=CCC(C)C(=O)NCCC1CC(OC)CN1C(c1cncc(CO)c1)=O Cc1csc(=O)n1CCCC(N1CCCC(CN(C)C(C2(C)CCCS2)=O)C1)=O c1(OC)ccc(C2(CNC(=O)C(N3CC(O)C(O)C3)c3cnsc3)CC2)c(C)c1 c1(C(N2CC(C)C(NC(c3cnn[nH]3)=O)C2)=O)cc2occc2n1C NC(CCC1CCCC1=O)CC(=O)NOCCC(F)(F)F.c1(O)ccccc1 CC(C)C1=NOC(C)(C(=O)NC(C)(C)CCNC(c2ccnc(C3CC3)c2)=O)C1 CN1CCCC1C=CC(N1CCN(C(=O)C(=O)Nc2cccnc2)CC1)=O C(=O)(C(C)(O)C(F)(F)F)N1CC(CN(C(C(C)CCc2cccc(F)c2)=O)C)C1 c1(OCC)cc(C(N2CC(=C(F)CNC(=O)C(C)OC)C2)=O)ccc1C c1(C(=O)NC(C2CCN(C(C(=O)NC(C)C)=O)C2)C)c(F)ccnc1Cl c1(C(N(C(C2(C(O)C(F)(F)F)CCC2)=O)CC)=O)cc(C)ccc1Cl N(C(=NCc1ccc2c(c1)CCCC2=O)N1CCC(O)C1)CCC(=O)NCC#C c1(COCC(=O)NCCC2(NC(C3(C(F)(F)F)CC3)=O)CC2)nc[nH]n1 CC(C)C(C(C)NC(=O)Cn1cnnn1)NC(c1cnc(C(N)=O)s1)=O c1(CC(N2C(CC(C(=O)N3C(C(=O)OC)CC3)F)CC2)=O)ncn(C)c1C C1(NC(CCc2n(C)cnc2)=O)C2CC1CN(C(=O)C(F)(F)c1cscn1)C2 N1(C(C2CCC3(CC3)C2)C(=O)NC(CC)C)CCCCC12CCN(C)C2 C1(NC(C(CC2CCC2)NC(c2cc(=NC)[nH]cc2)=O)=O)CC2CCC(C1)C2O C=CCC(C)C(C)(c1nnnn1CCSC)NCc1cc(C)n(C2CC2)c1C C(=O)(CCCOc1cccnc1)NCC(CO)NC(C1(CC=C)CC1)=O c1(CN(C(=O)CN2CC(C)(C(N)=O)C2)CCOCC#C)cccn1C C1(CC)CN(C(C2CCC3(CCC3)O2)=O)CCN1C(c1cn(C)nc1Br)=O N1(C(c2cccc(C#N)c2)C(=O)NC(C)C)CCc2ccc(Cl)cc21 Cc1nsc(C)c1C(=O)NCC(F)CNC(c1cccc(-c2cscn2)c1)=O CC1CN(C(=O)C(C)(C2CC2)N(C(=O)CC2COCCO2)C)CCN(C)C1 C1(CNC(N2CCC(c3ccc(C)cc3)CC2)=O)COc2ccc(F)cc2C1 N1(C(CC2(OC)CN(C(CN(CCOC)C)=O)C2)=O)CCOC(C)C1CO N1(C(Cc2cn(CC)nc2)=O)CC2(NC(=O)C(C(C)C)SC)CC1(COC)C2 CC1CC(N(C(=O)CN(CC(C)N(C)C)C)C)CC(C)(C)C1 Cc1ncc(C(N2CCC(NC(c3nc[nH]c3C(F)(F)F)=O)C2)=O)c(C(C)C)n1 N1(C(COC)=O)CCC2CN(C(c3ncc(C)s3)=O)CCC12 c1(C(=O)NC(C)CC(C)NC(c2cccc(O)c2F)=O)ccc([N+](=O)[O-])nc1 c1(C(=O)NCC23C(CN(C(CN(C)CC)=O)C2)C3)cn2c(n1)CCC2 n1(C(F)(F)F)nc(C(=O)NCC=CCNC(C2CC2(F)F)=O)cc1C1CC1 N1(C(C(COC)(C)O)=O)CC(CNC(=O)C(C)(C)n2ccc(C)n2)CC(C)(C)C1 C(C(F)CNC(=O)C(C1CCCC1)OCC)NC(COCCOCCCC)=O c1(C(=O)NCCN(C(=O)C=Cc2csc(C(F)(F)F)c2)C)cc[nH]c2nccc1-2 N1(C(CSCC=C)=O)CCC2(CCCC2CNC(=O)C(F)CC)CC1 N1(CC)C(=O)CCC1CC(=O)N(C(C)CNC(=O)COCC(C)C)C C12(NC(c3c(CC)n[nH]c3)=O)CCCC1N(C(c1ccc(O)c(OC)c1)=O)CC2 N1(C(c2cn(CCNC(C3CC3CO)=O)nn2)=O)CCC(O)C(F)C1 C1(CNC(C2(C#N)CCCC2)=O)CCN(C(C2CCC(=O)N2)=O)CC1O CCCCCCCCC(=O)N1CCCC(NC(=O)CCc2ccc(N)c(F)c2)C1 N1(C(=O)OC)CCCC1C(=O)NCC1(O)CN(C(C2COCCO2)=O)C1 c1(-n2c(C3C(C4N(C)CCC4)OCC3)nc(-c3cc[nH]n3)n2)ccc(C#N)cc1 c1(C(=O)NCC2COCCN(C(=O)Cn3cccn3)C2)cc2cc(Cl)cnc2o1 C1(C(N2CCC(NC(c3c(C)nc(C(C)C)s3)=O)C2)=O)CCC(C2CCC2)CC1 FC1(F)CC1C1CCCN(Cc2cnn3c2CCCC3)C1 C1(C(=O)NC(C)CC2CN(C(C3CC3C#N)=O)C2)CN2CCCC2CO1 C(=O)(C(C)C(=O)N1CC2(NC(=O)Cc3ccc(F)nc3)CC1C2)OC c1(NCC)ccc(CNC(N2C(C)CCC2C)=O)cc1 C1(C)(CNC(C=CCC)=O)CCN(C(=O)CCOCC2CC2)C1 N1(C(c2n(CCOC)ncc2)=O)CC2CC(NC(c3c(C)cnn3C)=O)C(C2)C1 N1(C(C(C)N(C)C)=O)CC(O)(CCNC(=O)C(C)C2CCCC2)C1 CC(C(=O)N1CCCc2nccn21)C1CCN(C(C2CC2(F)Cl)=O)CC1 c1(OC)ccc([N+](=O)[O-])cc1C(=O)NCC(C)N(C(=O)C1=C(C)OCCC1)C Cn1cnc2c1CCCC2C(=O)NC1CS(=O)(=O)CC1C(=O)O c1(CNC(=O)NCC(C)F)cc2sc(Cl)cc2[nH]1 c1(C(=O)NCC(CNC(c2c(NC)cnnc2)=O)OC)c(C)cccc1Cl c1(C(=O)NCC2(NC(C(=CC3CCC3)C)=O)CCOC2)ccc2[nH]c(=N)[nH]c2c1 c1(CC)oc2ccccc2c1CC(N1CCCC(CC)(NC(C2CCO2)=O)C1)=O C1(SCC)COCCN1C.C1(C2CCC2)C(=O)N1C1CC1.C12(CCC1)C(=O)N2.CCO N1(C(CC(C=C)CC)=O)CCC2(CCCC2NC(=O)COC2COC2)CC1 N1(C(c2c(S(C)=O)cccc2)=O)CC(C2CCCCN(C(=O)C3=CCCS3)C2)C1 C(=O)(C1=C(Cl)CCC1)N(CC(C)NC(=O)Cc1cccnc1Cl)CC CN=C(NCCCn1cccn1)N1CCC(Cc2ccco2)C1 C1(NC(C(C)(C)SC)=O)CCCC(NC(=O)COCC(C)(C)C)CC1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC)CCC2)=O)COCC(C)O1 N1(C(C(CC)C(C)C)=O)CC2CCN(C(=O)Cc3ccc(OC)cc3F)C2C1 C1(NC(C(C(C)C)SCC)=O)CN(C(=O)COC(F)F)C2(CCOCC2)C1 C1(NC(c2c(C)cncc2)=O)CCC12CN(C(=O)Cc1ccc(F)c(Br)c1)C2 N1(C(C(C)(C(=O)OC(C)C)OC)=O)CC2CN(C(=O)C(F)=CC3CC3)CC2(C)C1 N1(C(Cn2c(C)ccn2)=O)C(CC(=O)N(CC(C)O)C2CC2)C2CCCC12 C(C(C)(C)CC(=O)N(C(CC(C)C)C(=O)N(CC(F)(F)Cl)C)C)OC c1(C(=O)NCC2(NC(Cc3c(C)n[nH]c3)=O)CCC2)cccnc1O c1(C(=O)NCCCCNC(=O)COC2CC2(F)F)cc2cc(Cl)ncc2[nH]1 c1(C(N2CCC3C(C2)CN3C(=O)C#CC2CCOC2)=O)cnc2ccccn12 CC1CN(C(C2C(O)CCN2C(=O)C(C)NC=O)=O)C(C)C(C)(C)O1 C1(C2CC2)(CNC(c2c(C)cc(C)[nH]2)=O)CCN(C(c2cnn(C)c2Cl)=O)C1 c1(CC)[nH]ccc1C(N1CC(O)(C(F)CNC(=O)Cc2cncs2)C1)=O C1(C(=O)NCc2ccc(Nc3ncc(C(=O)OC)cn3)s2)CCC(C)=C(C)C1 N1(c2ncc(C(=O)OC)cn2)CCCC(C)(C(=O)NCc2ccc(Cl)c(Cl)c2)C1 N1(C(CCN(C(Cc2cc(C)no2)=O)C)=O)CC2=CCC(CC2)C1 n1(CCC)nc(Cc2ccc(OC)cc2)nc1-c1cnc(O)n1C c1(C(=O)NC2CC(CNC(c3nccc(OC)c3F)=O)C2)cnc2ccccn12 c1(CC(=O)NCC(C2CCCC2)NC(C(C)=C2CC2)=O)nc(C2CC2)n[nH]1 c1(C(=O)NCCC2CCN(CCc3nnn(C(C)C)n3)C2)cccc(F)c1 N1(C(C=Cc2ccc(C)o2)=O)CCC2(NC(c3nccs3)=O)CCCCCC12 N1(C(C(CC(C)C)N(C(C(C)OCC=C)=O)C)=O)CC2(CCOCC2)C1 C1(CC(=O)NC(C(C)NC(CC2(COC)CC2)=O)(C)C)C(=O)NN=C1C N1(C(C(CC)(CC)CC)=O)CCCC(C2CN(C(c3cccc(F)n3)=O)C2)C1 C1(C(N2CCC(N(C(C(C)=C(CC)C)=O)CC)C2)=O)CCC(C)(C)O1 C(=O)CCCC(C)=O.C12CC(C)N1C2=O.C1(=O)CN1C.CO n1(CC(=O)NC2CCN(C(=O)CCC3CC3)CC2CO)ccc2ccccc12 c1(C(N(C(C)CN(C(=O)C(F)C(F)(F)F)C)C)=O)ccc2c(c1)C(C)(C)CN2 c1(NC(=O)OCc2nc(C(=O)OCC)on2)ccc(Cl)c(C)c1 CN1CCC(C(N2CC=CC2CNC(c2ccsn2)=O)=O)CC1=O C=CCCCCCC(=O)N1CC(O)(CN(C(=O)CSc2ccc(O)cc2)C)C1 c1(CC(=O)NC2CC(F)(CNC(c3ccc(CC)[nH]3)=O)C2)ccc(F)c(Cl)c1F N1(C(C2C(C(=O)OC)CC2)=O)CC(NC(c2cc(C)nn2C2CC2)=O)CCC1C C1(NC(C(C)SCC)=O)CC(=O)N(C2CN(C(c3cocc3C)=O)C2)C1 N1(C(Cc2c(C)ncs2)=O)CC(NC(=O)CCc2cccnc2F)CC1(C)C c1(NC(C)=O)ccc(N)c(C(=O)NC2(CNC(c3ccnc(Cl)c3)=O)CCC2)c1 Cc1nc(C(C)C)ccc1C(=O)NC1CCC(NC(=O)CC2CCCCO2)CC1 c1(C(=O)NCC(C(=O)NC(CC=C)C)O)ncn(C)c1C C1(C(C)NC(=O)COCCF)CN(C(c2cc(-c3cnccn3)[nH]n2)=O)CCO1 C#CC1CCC(C(=O)N(C)CCN(C(=O)CCC2CCCO2)C)CC1 c1(CC(C)C(=O)NCC2CCN2C(=O)CCNC(=O)C=CCl)cccc(F)c1 C1(C(N2CCC(CNC(c3cnc[nH]3)=O)C2)=O)Cc2c[nH]cc2S1(=O)=O C(=O)(C(C(C)(C)C)NC(=O)COC1CC1)NC(C(C)C)CO C1(C(=O)NCCCN=[N+]=[N-])CCCCCN1C(=O)CCc1ccccc1 C1(NC(c2c(C)nccc2)=O)CC2C1CCN2C(c1ccc(C)c(O)n1)=O c1(CC(N2CC(CC(N3C(OCC)COCC3)=O)(OC)C2)=O)ccc(O)c(Cl)c1 C1(N(C2CC2)CC2(c3nnc(C)o3)CNC2)CCCCC1C Cc1cc(CNCc2cnn(C)c2Br)c(C)c(Cl)n1 C1(C(=O)NCc2c(C)cco2)CN(C(c2nnccc2C)=O)CCN1C N1(C(=O)NC2CCC2)CCN(Cc2ncc(Cl)cc2F)CC1C(F)(F)F c1(C(=O)NC2(C)CC(NC(CCCCOC)=O)C2)n[nH]c2c1CCOC2 c1(NCC(C)N(C(CCc2c(C)noc2Cl)=O)C)nc(C(C)(C)C)ccc1C#N c1(OCCC(N)=O)ccc(COC(=O)Cc2ccccc2N)cc1 c1(C(=O)NCC2OCCCO2)[nH]nc([N+](=O)[O-])c1Cl N1(Cc2nc(CC)sc2)CCC(C(N2CCCC(Cn3ccnc3)C2)=O)C(C)C1 c1(OC)ccc(C(=O)NCC2CC2C(=O)NCCC2CCC2)o1 C(CN1C(=O)Cc2ccccc21)NC(=O)C(C1CCCCCCC1)O Cc1nc(C)n(CCCC(=O)N(CCCCC2CN(C(=O)C3=NOCC3)C2)CC)n1 n1(CC)cnc2c(NCCN(C)C3CC3)[nH]c(=NCc3ccoc3)nc12 c1(C(C(=O)NCC2C(NC(C(C3CCOC3)OCC)=O)C2)(C)C)ccc(C)cc1 Cc1ccc(F)c(CC(N2CCCC(CNC(c3cc(CO)[nH]n3)=O)C2)=O)c1 c1(NCCN(C2CCCO2)C(c2ccc(N3CCOCC3)cc2)=O)ncncc1I CC1=C(C(=O)NC(Cn2cccn2)C(=O)Nc2ccc(C)nc2CO)SCCO1 CC1CN(C(=O)C2=NOCC2)CC1CNC(C1(n2cccn2)CCC1)=O c1(C(=O)NCC2C(NC(=O)C=Cc3ccccn3)CCCC2)cc(F)cc(Cl)c1 CC1C(NC2(Cc3cc4ccccc4[nH]3)CC2)CC2CCC1N2C N1(C(c2ccc(C(C)C)s2)=O)C2CCC1C(F)C(NC(=O)CN=S(C)(C)=O)C2 c1(C(=O)NCC2N(C(c3ccc(=N)[nH]c3)=O)CCC2)cn(CCO)c(=O)nc1O N1(C(CCC=C(C)C)=O)CC(NC(C2CC2(F)F)=O)C(C(F)F)C1 C1(NC(c2ccc(CSCCC)o2)=O)(CC)CCN(C(=O)C2=C(C)CCC2)CC1 C1(CC(=O)N(CCN(C(C(C)=O)=O)C(C)C)C)CCc2ccccc2C1 CC1CN(C(C2(C)CCCS2)=O)CC(C)N1C(=O)Cc1nc[nH]n1 c1(-c2cc(C(=O)OC)c(CO)cc2)ccc2nc(N3CCCCC(C)C3)sc2c1 CC1CCN(C(C2CCCN2c2ccccc2)=O)CC1NC(=O)CS(N)(=O)=O N1(C(C(CCNC(c2cc(C)c(O)nc2)=O)(C)C)=O)CCCNC(=O)C1C N1(C(c2[nH]cc(C(N)=O)c2)=O)Cc2occ(C(N3CCC4(CCC4)CC3)=O)c2C1 CCCCCCCCCC(=O)N1CCC(C(C)NC(=O)CCn2cccc2)CC1 N1(C(C(CC)OC)=O)C2CCC1CC(O)(CNC(=O)C(C(C)(C)C)NC(C)=O)C2 C1(NC(C(CCC)C(=O)OC)=O)CCN(C(=O)C(C)(C)CC)CC12CCC2 Cc1cc(C(=O)N(CCCN(C(=O)COCc2ncc(C)o2)C)C)cnn1 C1(C(C)C)N(C(c2ccncc2N)=O)CC12CCN(C(=O)C(C)(Cl)Cl)CC2 N1(C(COCCC=C)=O)CCN(C(=O)CN2CCC(O)CC2)C2CS(=O)(=O)CC12 C1(CNC(CSCC(C)C)=O)CC2CN(C(=O)Cn3ccc([N+](=O)[O-])n3)CC12 n1(CC(=O)NCC2C3CN(C(CC4(C)CC4)=O)C2C3)cc2ncccc2n1 Cn1cc([N+](=O)[O-])c(N2CC3CC(NC(c4cc(Cl)c[nH]4)=O)CC3C2)n1 N1(C(C2C(C)C2C)=O)CC2CCN(CC)CC2C1.N12CCC(CC1)C(=O)NC2=O C(CC(=C)C)(C(=O)N(C1CCCN(C)C1)C)NC(COCC#C)=O c1(C(N2CCN(C(c3cc(CCC)[nH]n3)=O)CC2C)=O)cc2ccc(Cl)cc2[nH]1 c1(C(=O)NC2CN(C(c3ncc(CC)nc3)=O)CC3C2C3)cn2nc(C)sc2n1 c1(OC(COC)C(=O)NCC(C)CN(C(=O)C(C)(C)C)C)ccc(F)cc1Cl C(C)(C(=O)OC)N(CCC)C(C1(c2cc[nH]n2)CC1)=O.C1(C)CCC1 N(C(=NCCCCC(F)(F)F)NCC1CC2CCC2C1)C1CC(OC)C1 O=C1CC(C(=O)NC2CCCCN(C(=O)C(F)CC3CC3)C2)NC(=O)N1 C(=O)(C1=C(C)OCC1)N1CC(NC(C(CC)n2cccn2)=O)C(SC)C1 C12(NC(c3cnc[nH]3)=O)CC3CC(C1)CC(NC(C1CC=CCC1)=O)(C3)C2 CCC(O)CC(=O)NCCCC(C)NC(c1ccc(-c2cnn(C)c2)cc1)=O C1(C(=O)NC(C=C)CO)CC(O)CCN1Cc1ccc(N2CCOCC2)s1 c1(CNC(c2n(CC)ccc2)=O)ccc2c(c1)CCN(C(=O)Cc1cocn1)C2 n1(CC(=O)NC2C(NC(C(CC)OC)=O)CCC2)ncc(Br)c1C C1(CNC(C(CC)N(C)C)=O)CC(C(=O)Nc2ccc(O)c(OC)c2)=NO1 CC(O)CCC(=O)NCCC1CSCCN1C(c1cc(C(F)F)ccn1)=O C(CCC)(CCCNC(c1ccc(CC)cc1)=O)NC(C=CC(CC)=CC)=O C1(CNC(C2(NC(C3CCN(CC)C3)=O)CC(O)C2)=O)CCCCC1(C)C N1(C(C#CC(C)C)=O)CCC2(CCCCC2NC(=O)COCCCF)CC1 N1(C(CC(=C=C)C)=O)CCN(C(c2cccnc2O)=O)C(CC(F)(F)F)C1 Cc1cc(NC(C2CC2)=O)ncc1NCCN1CCOCC1 N1(C(c2ccc(OCC#N)cc2)C(=O)NCC=C)CCc2cc(Cl)ccc2C1C Cn1cc(CCC(=O)NC2(CCO)CN(C(=O)C=CC3CCCO3)C2)cn1 N(C1CCc2ccccc21)(CC(c1ccc(O)cc1)=O)C(C)=O CCC(CNC(c1ccc(N)cn1)=O)(CC)NC(=O)C(COC)c1ccccc1 C(N=c1[nH]c2c(c(=NC(C)CC3CC3)[nH]1)CCCCCC2)C1(COC)CCOC1 N#CC1CN(C(c2cc(-c3ccccc3)cnc2O)=O)CCO1 c1(OC)ncc(C(C(=O)NC2CCCC2)N(C)CC2CCCC(C)C2)cc1Cl CC(C)(C#N)CC(=O)N1CCC(CC(=O)NC2(C(C)(F)F)CC2)CC1 N1(C(C2C(OC)(OC)CC2)=O)CCC(F)(CNC(C2CCC(C)(C)C2)=O)CC1 c1(C(c2nnnn2CC(F)F)N(CCCO)CC2CCC2)ccc(Cl)c(Br)c1 CC1CN(C(=O)C(C)C(F)(F)F)CCCN1C(c1c[nH]c(C(N)=O)c1)=O c1(-n2cc(CN(C(c3c(C)nc(CC)o3)=O)C)nn2)ccc2c(c1)CCCC2 Cc1sccc1C(=O)NCc1ccc(C2(N)CC2)o1 c1(N(CC(F)(F)F)C(c2cccs2)=O)ccc2ccccc2c1 C(C)(C(=O)N(C)CCNC(=O)C(F)=CCC)OCCC=C CC1(C)CC(C(=O)NC2CC(CCNC(C3CC(F)C3)=O)C2)CC(C)(C)O1 CCC(C)C(=O)C(=O)NOCC(=O)Nn1cnnc1O C(=O)(C1=C(Cl)CCOC1)N1CCC(CN(C(c2cnc(C)n2C(F)F)=O)C)C1 C1(CNC(COCC)=O)CC2(CCC2)CN1C(=O)C(CC)(CC)c1ccccc1 C(C=CC(=O)NCC1CCC1NC(=O)C=CC(=O)NCC1CC1)(CC)=CC N1(C(C(CC=C)C)C(=O)Nc2ccc(OC)cc2C)CCN(C)C2(CCOC2)C1 C1(NC(C2(N(C)C)CC2)=O)CCNC(=O)CC1.C12CCC(CC1)CNC2=O C(=O)(C(CC)CC)NCC1CC(F)(CNC(C=C(CC)C)=O)C1 C(=O)(CC(C)(C)C(=O)OC)N(CCNC(C1(CC#C)CCCC1)=O)CC N1(C(C(c2cn(C)nn2)NC(C(CCC(C)C)=O)=O)=O)CCc2c(nnn2C)C1 CCC(C(=O)NC(C)CN(C(c1nncn1CC)=O)CC)C(C)C C1(CCN(C(CC)C2COC2)C(c2cccs2)=O)CC2(CCN(CC(C)(C)C)C2)C1 c1(-c2ccc(C#N)cc2)cc(C(=O)Nc2cnc(F)c(Br)c2)c2cn[nH]c2c1 N1(C(C2N(C(C)=O)CSC2)=O)CCOCC(NC(c2nocc2C)=O)C1 c1(NC(=O)NCCCCSc2ccccc2)ccc2c(c1)CCO2 c1(C(C(c2nnnn2C2CCOCC2)NC(C)CCCO)(C)C)ccc(Br)cc1 c1(C(=O)NCCOCCOCCCNC(CC(=C)C)=O)ccc(C)c(C(C)=O)c1 N1(C(c2c(CC)cno2)=O)CCC(F)(CNC(=O)CCC2CCC(=O)N2)C1 N1(C(CNC)=O)CCCC(N2CCCCC2)C1.c12ccc(cc1)C1(COC1)NC2 C(C)(C(=O)N=c1cc[nH]cc1)NC(c1cc(Cl)cc(Cl)c1)CC Cc1cc(Cl)ccc1C(=O)NC1CCC(C)N(C(=O)CCC=CBr)C1 c1(C(=O)NC2C3CN(C(C(c4c(Cl)cnn4C)C)=O)CC32)cc(Cl)c(F)cc1O C1(CC(=O)NCCN2CCOC2=O)CCCCN1C(c1cc(Cl)n[nH]1)=O C1(NC(C2CC(CC)C2)=O)COCC1C(=O)NCC1CCOC1C C=CCCCC(=O)N(C)CC1(NC(=O)CN2CCC(F)(F)C2)CC1 C(=O)(C(F)C(C)C(C)(C)C)N1CCC2(CN(C(c3ccc(OC)s3)=O)C2)C1 C(=O)(CCCN1CCCC1)NCCN(C(c1c[nH]nc1C1CCCO1)=O)CC c1(C(=O)NCC2C(C(N3CCCN(C(=O)OC)CC3)=O)C2)cc(Cl)c(Br)cc1Cl N1(C(c2c(CC)cc(N)cc2)=O)CC2CC(NC(=O)CCC(C)C)CC1C2 c1(C(=O)NC(CC)CNC(c2ncccn2)=O)cc(Cl)cc(C)c1OCC(N)=O C(c1ccc(Cl)cc1Cl)=CC(N1CCCC(CNC(=O)COCC(F)F)C1)=O C(=O)(C1=NOC2COCC12)N1C(C)CC(NC(C2(C)CC(=O)C2)=O)C1 Cc1cnc(C(=O)NCCC(C)N(C)C(C2CC2c2n[nH]c(C)n2)=O)nc1 c1(OC)cc(C(N2CCC(F)(C(N3CCCOC(C)C3)=O)C2)=O)cc(OC)c1Br C1(C(N2CC(=C(CNC(CC3CC(C)(C)OC3)=O)F)C2)=O)CCCC(F)(F)C1 c1(CC(=O)NC2CC(NC(CCC(C)(F)F)=O)C2)coc2cc(Cl)ccc12 C1(CNC(CCC(C)(C)N2CCOCC2)=O)CN(C(=O)CO)CC12CCOCC2 N(C1CCc2ccc3c(c21)CCO3)C(c1ccc(C(C)C)c(Cl)c1)C N#Cc1cc(C(=O)NCC(=O)N(CCCF)CC(N)=O)cs1 c1(OC(C)C)ccc(C(=O)N(C(CNC(=O)C#CC2CC2)C2CC2)C)cn1 c1(NCCCCNC(C2(COC)CC2(F)F)=O)ncn(C)c(=O)c1Br C#CCCCC(C)C(=O)NC1(CCCNC(C2CC2CC)=O)CC1 Cc1cc(C(=O)NC2CC(C)CN(C(=O)CC3CCS(=O)(=O)CC3)C2)cnc1C c1(CC2C(C(N3CCOCC3C3CCCC3)=O)CCCC2)cc2n(n1)CCCC2 c1(NC(=O)NCCCC2(O)CC2)sncc1Br c1(C(=O)NC(C2CCCOC2)C)n[nH]c2c1CN(C(=O)CN1CCC(F)CC1)C2 c1(C(=O)NC2C(CC)CN(C(C3(CC)CC3)=O)CC2)cc(=O)n2ccsc2n1 Nc1c(C(=O)NCCC(O)CNC(=O)CC2CC2(Cl)Cl)cnn1CCO C1(CC=C)(NC(=O)C(c2cscn2)N(C)C)CCN(C(c2ccc(=N)[nH]n2)=O)C1 C1(C(N2CC(CC)(NC(C3CCCN3C=O)=O)C2)=O)CC(=O)CC12CCC2 N1(C(C(C(C)O)(F)F)=O)CC2CCCC2(CNC(=O)Cc2cn(C)nn2)C1 CC1CCN(C(C2CN(C)C(=O)N2)=O)C(C)C1NC(=O)Cc1cccc(Cl)c1 c1nn(CC2CC2)cc1C(c1nnnn1CC1CC2CC2C1)NC1CCOCC1 C1(C(=O)NCCNC(Cc2c(OC(C)(C)C)cccc2)=O)CCCN2CCCC12 CCCCCC(CCC)C(=O)N1CC2C(CNC(=O)CC3COC(=O)C3)C2C1 c1(C(c2nnnn2C2CCOC2)(C)Nc2c(CC)ccs2)ccc(C(C)C)cc1 c1(CC)cnoc1C(=O)NCCN(C(c1cc(COC)on1)=O)CC1CC1 c1(C(=O)NC2C(C)N(C(c3cn(C)nc3C(F)F)=O)CC2)cccn(C2CC2)c1=O C1(C(N(CCC(=O)NC)CCO)=O)(NC(=O)CCSC)CCCC1 C(=O)(CCCN=[N+]=[N-])NC(C)C=CC(=O)Nc1cccnc1 c1(OC)ccc2c(c1)C(C(=O)NC(C)CCNC(C1(C(=O)OC)COC1)=O)CC2 N1(C(CC(C)(C)OC)=O)CCCC(C)(C(=O)NC(c2cscn2)CO)C1 N1(C(C(C=C)O)=O)C2CCC1CN(C(=O)Cn1cnc(C#N)n1)CC2 c1(CNC(c2ccc(C)cn2)=O)nc2c(s1)CCN(C(=O)C(C)OC1CCCC1)C2 C1(CO)CCCCC1.c1(C(=O)NC(CC)C(N)=O)cc(CN)nn1C C1(CC)C(C(=O)NCC(F)(F)C(N)=O)CCCN1C(c1cnc[nH]c1=N)=O N1(C(c2ccc(CC)[nH]2)=O)CCN(C(=O)CCS(C)(=O)=O)C2CC12 CC12CC(C(=O)NC3CCN(C(C4CCN(C5COC5)C4)=O)C34CC4)(C1)C(C)(C)O2 N1(C(C2C(CC)(CNC(CC(C)(C)COC(C)C)=O)C2)=O)CCCC(CC)C1 CCCC(C)CC(=O)N(CCCC(=O)NC1CCC(C)(O)CC1)C C1(S(N)(=O)=O)(C(=O)NCCN(C(=O)CNC(=O)CCC2CCCC2)CC)CC1 C#Cc1ccc(C)c(NC(C2C(C)CCN2C(c2nnc(S)n2C)=O)=O)c1 C1(N(C(C(CN(CC)CC)F)=O)C)CN(C(c2c(O)cccc2Cl)=O)CC12CC2 c1(NC(c2ccc(C(C)(C)C)cc2)C)c(C)c([N+](=O)[O-])ncn1 O=C(C#Cc1ccccc1)N1CC2CCC1CN2Cc1ccc(CO)o1 C1(C(N2CC(c3cn(C4CCOC(C)C4)nn3)C2)=O)CCOC(=O)N1 N12CC3CN(CC(C1)O3)C(=O)C2=O.c1(C(=O)OCC)cn2cc(Br)ccc2n1 C1(NC(C(CC=CC)NC(=O)CC2CCCC3CC23)=O)CC2C(O)C(O)CC12 CCCC(C(=O)OC)C(=O)NCC1(CCNC(=O)C(C)Cc2cnc[nH]2)CC1 c1(CNC(CCN(CC#C)C(c2cnn(C)c2CC)=O)=O)cc(C)cc(F)c1 Cc1cnc2n1CCC(C(=O)NNC(=O)N1CCN(CC(C)C)CC1)C2 N1(c2nc(SC)nc(C)c2Br)CCC2(C1)OCC1CC21 CC1CC(C(=O)NC(CCCN(C)C(c2ccc(NCCO)cc2)=O)C)=NO1 C(C)(C(C(=O)NCCc1cscn1)C(C)C)NC(C(=O)NC(C)C)=O C(=O)(CC(CC)SC)N(CCNC(C1(CCC=C)CC1)=O)C1CC1 C1(O)(CN(C(c2c(C)csc2)=O)C)CCCN(C(C2CCNC(=O)C2)=O)C1 CC12CCOC(C(=O)NCC(F)CNC(c3ccnn3CC(F)(F)F)=O)(C1)C2 c1(CC)cc(F)ccc1C(N1CCC(NC(C2CC=CC2)=O)C(CC)C1)=O Cc1ccc2ncccc2c1C(=O)NCCN(C(=O)C1=CC(C)(C)C1)C1CC1 C1(O)(C(C)NC(CCC#CC)=O)CCN(C(C2CC2c2ccoc2C)=O)CC1 C1(C(=O)NC2CC(O)(CC#C)C2)CCC2CCC1N2C(c1c[n+]([O-])c(C)cn1)=O c1(NC(CCSC)C)ncc(S(=O)(=O)NC(c2ccc(F)c(C)c2)CO)cc1Cl CCCCC(O)C(C)C(=O)N1CCC(F)(C(=O)N(C2CC3CC3C2)C)C1 c12cc(cc(C(C)C)c1)OC2=O.CCCCN(CC(F)F)C#N N1(C(CC2(O)CC(C)(C)OC2)=O)CC2CCC1C(Nc1ncc(C#N)cc1Cl)C2 Cn1cc(C(=O)NCC(C2CCCC2)NC(C2(C(F)F)CCCO2)=O)cn1 N1(C(Cc2nc(C)sc2C)=O)CC2(CCN(C(=O)C=Cc3cccc(O)c3)C2)C1 c1(C(N2CC(c3cn(C(C(=O)OCC)C)nn3)C(O)C2)=O)ccc(F)cc1SC c1(NC(C2N(C(c3c(C)cccn3)=O)C3C(C2)C3)=O)ccc(Br)cc1C#N C(C)(CO)(CC(F)F)N(C(c1cc(OC)ns1)C(=O)NCCOC)C C1(C(N(CC(CNC(c2scc(C)c2Cl)=O)(C)C)C)=O)CC2OC(=O)OC2C1 CCC(CN(C)C)CC(=O)N1CCC(N2CCC(NC(=O)C(C)(C)C)CC2)C1 CC(C)(C)C(CC(=O)NCC(O)CNC(c1cc(Cl)cc2c1OCC2)=O)C(F)F C(=O)(CCCCC(=O)N1CCCC(C(C)NC(=O)Cc2ccn(C)n2)C1)OC Cc1cc(NC2C(C)CN(C(c3ccn(C(C)C)n3)=O)CC2C)n2nnnc2n1 N(C(=NCCN1CCC1)NCC(=O)N1CCCC1)CC1C(C)(C)CCO1 Cc1cc(CC(N2CCC(NC(=O)Cc3ccc(F)cc3)CC2)=O)n(C)n1 C1(=O)CCCCNC(=O)CN1C(C)=O.C(CN(C)OC)N.CCCS C1(NC(C(CC)(C#N)CC)=O)CCC2(CCCN(C(=O)C3=NOCC3)C2)C1 Cc1ncc([N+](=O)[O-])n1CCCn1cccc1 CC1CN(Cc2ccc(F)cc2)CC1NCc1cn(C)c(-c2ccccn2)n1 C(C(=O)NOCCN(C)C)(c1cn(C)nc1)NC(=O)COC1CCCCC1 c1(C(=O)NCC2C(NC(CC(=C)C)=O)COC2)cn(C)nc1SC CCC(CC)C(F)C(=O)N1CCC(C)(CNC(=O)CCc2ccncc2)C1 c1(C(=O)NC(CCC)CNC(C23CCN(CC2)C3)=O)cnc(C)nc1C(C)C C1(CC(=O)NCCC2CCN(C(c3cc(OCC)cs3)=O)C2)(CC=C)CCCC1 C1(C(=O)NCC2N(C)CCN(C(Cc3c(C)con3)=O)C2)CNC(=O)C(C)(C)C1 N=c1[nH]c2c(s1)CCCC2C(=O)NCC(F)CNC(c1ccn2ccnc2n1)=O Cc1cccc(F)c1C(=O)NC1CCCN(C(C2(c3cccnc3)CC2)=O)CC1 N1(C(=O)C=CCn2cncn2)CCC(CF)(NC(c2cc(C(F)F)[nH]n2)=O)C1 C(=O)(CN=c1[nH]c(=NCc2cn(CC(C)(C)C)nn2)c2ncccc2[nH]1)NCC=C Cc1cc(=NCC2(C)OCCO2)[nH]cc1S(=O)(=O)N1CCC(N)C(C)C1 C(=O)(C1=CCCSC1)NCc1cccc(C(N2C(CC(C)C)CCC2)=O)n1 C1(C(N(C2CCN(C(=O)C(=Cc3cnc[nH]3)C)C2)CC)=O)CCn2nnnc2C1 N1(C(CC(=C)C)=O)CC2(C1)C(NC(C1CCCC3C1C3(F)F)=O)CCS2(=O)=O c1(N(CCC)CCNC(c2n[nH]c(C3CC3)c2C)=O)ncnc2scnc12 N1(C(=O)CC2CCC=CCC2)CC2CC1CN2C(=O)COC1CCC1 CC1CN(C(=O)COCc2nc[nH]n2)CCC1NC(C1CC(=O)N(C2CC2)C1)=O c1(C(=O)NCC=CCNC(C(C)OC)=O)cc2c(nn1)CCCO2 C1(NC(CCC(C)NC(=O)CCn2cnc(=N)[nH]2)=O)(CO)CC2(CCC2)C1 c1(C(N2CC(C)C(NC(=O)C=CC(=O)NC3CC3)C2)=O)cncc2cccnc12 N1(C(CCn2ccc(=N)[nH]2)=O)CCCC2(CCCN2C(C2CC3CC3C2)=O)C1 N1(C(CC2CCN(C(c3[nH]cc(C)c3)=O)C2)=O)CCOC(C(C)C)C1 c1(SCCC(=O)NCCN(C(=O)C(c2ccc(O)cc2)=O)C)ccccc1Cl Cc1cnc(Cl)c(CN2CC3C(C(N4CCCC4c4ccccc4)=O)C3C2)c1 C=CC(C)(O)CC(=O)NC1CCOC1C(N1CCC(OC2CC2)CC1)=O C1(OC)CCCN(C(=O)NC2CC3CCC2C3NC(=O)OC(C)(C)C)C1C C#Cc1ccc(NC(=O)Nc2cc(Cl)c(Cl)c(Cl)c2)nc1F C12(C(=O)NCC3OCCN(C(COCCOC)=O)C3)CCCC(CO1)C2 CCC(C(=O)NCC(C1CC1)NC(c1oncc1C)=O)C(C)C C1(CNC(c2nc(Cl)cs2)=O)CN(C(C2CC(=O)N(O)C2)=O)CCCO1 N1(C(c2cc(SC)oc2)=O)CC2CC2(C(=O)NC2CCN(C)C2=O)C1 c1(C(C(=O)NCC=C)N(C)Cc2cccc(OC)c2F)nc(Br)ccc1OC C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)CCc2cncnc2)C12CC2 C1(C(N2C(CNC(C(C)(C3CC3)NC(C)=O)=O)CC(O)C2)=O)CCCN1N=O C=CCCC1C(=O)N1.c1(C(=O)OC(C)(C)C)ncc(C#N)o1.C1CS1 C1(CC)C(NC(c2cc(SC)n(C)n2)=O)CCN1C(=O)Cc1cc(C)[nH]n1 Cn1cc(CC(=O)NC2CC(C(C)NC(c3cccs3)=O)C2)cn1 c1(NC(c2nnnn2C2(C)CC2)C2(CSC)CC2)cncc(F)c1 C1(CNC(C2(CC#C)CCCC2)=O)CCCCN1C(=O)CCCCNC(N)=O Cc1ccc(CCCNC(=O)NCC(C2CCCC2)N(C)C)s1 c1(CNC(C(C)OCC)=O)ncoc1C1CN(C(c2nc[nH]c2C(C)(C)C)=O)C1 C=C(F)C1(CC(=O)NC(C(=O)NCC2CC(OCC)C2)C(C)C)CCCC1 N1(C(CC=CCC)=O)CCC(CCNC(=O)Cc2cc(C)on2)C(F)(F)C1 C(C(=O)O)(C(CO)C1CC1)OC.c12ccccc1OCC(=O)N2 c1(C(=O)NC2C(NC(=O)Cc3ccsc3)CCC2)cccn2cncc12 Cc1c(C(N2CCCC(N(C(=O)COC3CC3)C3CC3)C2)=O)ccn1C(C)C N1(C(C2N(C)CC(O)CC2)=O)CC2COCC2(C(=O)NCC2CCCC2)C1 c1(C(=O)NCC(C2CCN(C(CN(C(C)C)C)=O)CC2)C)ccc(C#N)c(Cl)c1 Cc1cc(C)c(C(N2CCN(C(c3coc4c3COC4)=O)CC2)=O)c(C)c1 c1(N(C(CCOC(C(C)NC(CS(CC)=O)=O)=O)C)C)nc2cccc(C)c2s1 S(=O)(=O)(c1ccc(NCC2CC(F)(F)C2)cc1Br)NC(c1c(C)nc(CC)o1)C c1(OC)ccc(CN2CC(NC(=O)C(=O)NCc3ncc(Cl)s3)CC2=O)cc1 Cc1c(CNc2cn(C)c(C(=O)Nc3ccc(Br)cc3F)n2)ccnc1Cl N1(C(c2onc(C)c2C)=O)CCCN(C(c2ccco2)=O)C(C(C)C)C1 C(=O)(C1Cc2cccc(Cl)c21)NCCC1CCN(C(CSCC(C)C)=O)CC1 C(=O)(CCS)N(CCC#C)CCC.C(=O)(CN(C)CC)N(CCO)C(C)C C(=O)(C#CC1CCCCC1)NC1CCC(NC(c2c(CC)cc[nH]2)=O)C1 C1(C(N2CC3C(NC(CC(=C)C)=O)(C3)C2)=O)CCCCC(F)(F)C1 c1(C(C)C(=O)N(CCNC(c2cnc(C3CC3)s2)=O)C2CC2)ccc(F)cc1 C1(C(=O)NC(C(=O)NCCc2c(C)n[nH]c2)CC2CCC2)CCC(C)(C)CC1 C1(C(=O)NCC2N(C(c3c(CC)scc3)=O)CCCC2)(CC)CCC(O)CC1 C1(C(=O)NCC(COC)(C)O)C2CCN(C(C3(OC)CC3)=O)CC12 c1(CC(=O)NCC23OCC(NC(C(C)(C)O)=O)(C2)C3)cccc(Cl)c1C(F)(F)F c1(C(=O)NC(CN(C(c2c(Cl)cc(C)c(N)c2)=O)C)C)cccc(Cl)c1[N+](=O)[O-] Cc1cc(=NCC2CNC(=O)C2)[nH]cc1S(=O)(=O)N(C)Cc1ccc(Cl)c(Cl)c1 N1(S(c2c(C)oc(CO)c2)(=O)=O)CCC2(CCCC(C(=O)O)O2)C1 c1(CC(N2CC(OC)(CNC(=O)C(C)n3cccc3)C2)=O)ccc(C2CC2)cc1 C1(C)(CNC(C=CCOC)=O)CCN(C(=O)C(C)Oc2ccccc2)C1 C(=O)(C1=CCc2ccccc21)N(CC(CN(C(C(C(C)C)SC)=O)C)O)C c1(CC(N2CC(CNC(C3CC(OC)C(OC)C3)=O)C2)=O)nsc2ccccc12 CC1CC(NC(=O)C(C)(C)C)CN1C(=O)CSCC(N)=O.C1(=O)NO1 c1(OC)ccc(C(O)C(N2CCC(C)C2CNC(=O)C#CC(C)C)=O)cc1 CCCCCC(O)CC(=O)N(C(C)CNC(c1cccn(O)c1=O)=O)C Cn1ncc2cc(CNC3CC(C(=O)Nc4ccc(Br)nc4Cl)C3)ccc12 CC1(C)C(NC(=O)Cc2ccoc2)CC1CNC(=O)CN1CC(=O)NC1=O c1(C(N2CCC(CNC(C(C=C)(C)CC)=O)C2)=O)cn2c(Br)cccc2n1 C1(NC(=O)NC)COCC1n1cc(C)nn1.C1(COC)(OC)CCOC1 C1(C(N2CCC(CSC)CC2)C(=O)OC(C)(C)C)CC(C)CC(C)C1 N1(C(c2c(C)nsc2C)=O)CCC2(CC1)CC2C(N1CC2(CNC(=O)N2)C1)=O C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CC(C)NC(c2ccoc2Cl)=O)CC1 C1(NC(c2c(C)nc(C)o2)=O)CC2CC1N(C(=O)C=Cc1nc(C)cs1)C2 C1(C(=O)NCCN(C(=O)CCN2CCC(F)C2)CC)(CC)CCOC1 c1(CC(N2CCCC(CNC(CC(C)C)=O)C2)=O)c(F)cc([N+](=O)[O-])cc1F c1(CC)c(C(=O)NCCC2(NC(=O)Cn3cc(C4CCOC4)cn3)CC2)nnn1C C12(CNC(=O)C=CCO)CC1CN(C(c1ccccc1Br)=O)C2 C1(C(C)NC(=O)C(=O)NC(c2ccoc2)C)CCC(C(F)F)CC1 c1(C(N2CC3CC3(C(=O)NCCc3ccc(O)cc3)C2)=O)cccc(Br)c1Cl N1(C(c2cncc(CNC(C3C(C)(C)C3(C)C)=O)c2)=O)CCC2(CCOC2=O)C1 C(C(C)(C)C#N)NC(C(C1(C)CC1)NC(COCCOCC)=O)=O C=C(C)CCCC(=O)NC1CCCN(C(=O)CC(CC)C2CC2)C1CC n1(CC)cc(CN(C(=O)CC2CCCN2C(c2cnsc2C)=O)C)cn1 CCC(C)CCCCC(=O)N(CC(C)(C)NC(=O)C1=CCCCC1)C c1(C(=O)NCCCC(C)NC(CCC=C(C)C)=O)cccc(C(=O)OC)n1 c1(NCc2nnn(CC)n2)ncc(S(=O)(=O)NCC(C2CCCC2)O)cc1Cl CC1(C)CN(C(=O)CC2OCCO2)C(CNC(c2cccc(Cl)c2)=O)CO1 C1(C(C(N2CC(N(C)CC)C2)=O)C)CCN(C(C2(C)CC2C)=O)CC1 C#Cc1cc(C(=O)NC2CCC(N(C)C(c3c(C)cccc3Cl)=O)C2)cc(N)c1 C(N=c1nc(C)[nH]cc1C#N)C1CC(NC(C(C)NS(CC)(=O)=O)=O)C1 C=CCCC(C)(C)C(=O)N(C)CCOCCC(=O)NC(C)C(C)SC C#Cc1cn(C)nc1C(=O)NCC1CCCCCN1C(=O)CC1CC1C(F)(F)F c1(NC2CCN(CC)C2)cc(N2CCN(c3cc(SC)ncn3)CC2)ncn1 c1(C(N2C3CN(Cc4ccncc4O)CC23)=O)ccc(-n2ccnn2)cc1 C1(C(=O)NCC(CNC(c2ccn(CCF)n2)=O)CO)(CC)CC1(F)F c1(C(=O)OC)cccc(C(=O)NCCNC(C2CC(F)(F)C2)=O)c1C N1(C(c2scc(C)c2)=O)CCc2cc(CO)ccc2C1.N12CCCC(C1)C2=O C(CCCC(=O)N1CCCC(CCF)C1)NC(c1n[nH]cc1Cl)=O C(C(C)CC(=O)NC1CCCCC1CNC(=O)Cc1csc(S)n1)OC C(=O)(C1=CCC2CCC1N2C(=O)C(C(C)C)SC)NCC=CCCC N1(C(CNC(Cc2cccc(OC)n2)=O)=O)CC2CC1CN2C(c1cnoc1C)=O CC(O)(C(=O)NCCCC(c1ccccc1)NC(C1CC2(CC2)C1)=O)C1CC1 N1(C(c2cnc(CCCC)s2)=O)CCC(CNC(=O)CC(=O)N(C)C)C(C)C1 C(=O)(C(CCCC)NC(c1ccc(C(F)F)o1)=O)NCC(CC=C)(F)F c1(OCC)nc(N2CCC(CNC(=O)Cc3c[nH]nc3C)C2)ncc1C CC1(C)CCC2(CC1)CC2C(=O)NCCC1=CCCCCC1 C1(F)(CN(C(=O)NCc2cc(N3CCOCC3)ccn2)C2CC2)CC12CCCCC2 C1(C(=O)NCC(C)(C2CC2)NC(=O)CCn2ccccc2=O)Cc2nncn2C1 c1(C(=O)NCC2N(C(C3CC(=O)NC(=O)N3)=O)CCOC2)cc([N+](=O)[O-])ccc1Cl N1(C(c2cn(C)c(=O)n2C)=O)CCCC12CCN(C(=O)Cc1cncs1)C2 Cn1c(Br)cnc1S(=O)(=O)NC(C12CC1CCCN2)Cc1ccccc1 N1(C(c2c(OC)csc2)=O)CCC(C)C(C(=O)NC2(CO)CC=CC2)C1 c1(C(N2CC(NC(Cc3ccc(SC)s3)=O)C2)=O)cc2c(=O)[nH]ccn2n1 C1(NC(=O)CC2CC2)CCCC(NC(c2noc(Cc3ccc(F)cc3)n2)=O)C1 c1(CCNC(CN(C(C=CC(CC)C)=O)C2CC2)=O)ccnc(C)c1 CCCCC(C)(F)C(=O)NC(CC(=O)N1CC2CC2C2CC12)CC(C)C Cc1nocc1CC(=O)NC(C1CCN(C(c2ncsc2C(C)C)=O)C1)C C1(NC(C2(C)C(C)(C)C2)=O)C=CCC(C(=O)NCCc2cocn2)C1 CCC(CC(=O)NC(CC1CC1)C(=O)NCc1ncsn1)C1CC1 CCC(C)(COC)C(=O)N(C1CCN(C(C2COCCN2CC(F)F)=O)CC1)C c1(C(=O)NCCCC)csc(C2CCCN2C(c2ccc(C)s2)=O)n1 C1(=O)C2C(CNC(=O)N(CCOCC)C(CC)CC2)N1 N1(C(C(CC#C)C)=O)CC(NC(=O)C#CC(C)(C)C)C(S(C)(=O)=O)C1 C1(CC(=O)NCCC2(CNC(CCOCC#C)=O)CCC2)CCC2CC12 c1(CC(N2CC(CN(C(CCN(C(C)=O)C)=O)C)OCC2)=O)ccc(O)c(O)c1 c1(C(=O)NC2(CNC(C(C(CC)C)O)=O)CCCCC2)cccc2sccc12 N1(C(c2c(CC)nn(C)c2)=O)CCCCCC1C(=O)NCCN1CCCC1=O C1(CC(N2CC(O)(CNC(C(C)CC3CCCC3)=O)C2)=O)CCCC2(CCC2)O1 N1(C(CN(C(C(C)n2ccnc2)=O)C2CC2)=O)CC(C)=CC(C)C1 c1(C(=O)NC2CC3CN(C(c4ccccc4Cl)=O)CC23)cnc2ccccn12 CC1CN2CCN1C(C(N1CC3C(CNC(C4(N(C)C)CC4)=O)C3C1)=O)C2 c1(C(N2C(CNC(C3C(C)C3C)=O)CCCCC2)=O)ccc2ccccc2c1 C=C(C)CC(C(=O)N1CCN(C(c2cncc(F)c2)=O)C(CF)C1)NC(C)=O Cc1ccc(CNC(c2ccc(C)c(Br)c2)C)c(O)c1 Cn1ncc2c1C(Nc1cc(N3CCCC(C(N)=O)C3)ncn1)CCCC2 CC(F)(F)C(F)(F)CC(=O)NCC1CC1CNC(=O)C1=CC2C=CC(C1)C2 CC(CNC(c1ncccn1)=O)CC(=O)NC1CCCN(C)C1 CCCCCCC(CC)C(=O)NC1CC(NC(=O)C=Cc2ccc(Cl)cc2F)C1 S(=O)(=O)(c1cccc(=NC(C)CC(C)O)[nH]1)NCc1c(C)ccc([N+](=O)[O-])c1 CCCC(CC(C)C)C(=O)N1CC2(C1)CN(c1ccc(C#N)c(C3CC3)n1)C2 Cc1cc(C(=O)NC2CCC(CCC(=O)NC(C)CCC3CCCC3)C2)cc(C)c1 c1(SC)cc(C)ccc1C(N1CCC(CNC(=O)C(C)OC2CCCCC2)C1)=O c1(C(=O)NC2CN(C(CCSC)=O)CC(O)C2)c(Br)nc2n1CCC2 N1(C(CC(Cc2c(OC)cccc2)C)=O)CCC2CCN(C(=O)C=C3CC3)C2C1 c1(C2CCN(C(C(CCCC)Br)=O)CC2)nsc2ccccc12 C1(CC(=O)NCCC(CC)C)CN(C(=O)Cc2ccc(O)cc2)CC12CC2 Cc1cc(=NC2CN(C(c3ccc4nsnc4c3)=O)CC2C)c([N+](=O)[O-])c(C)[nH]1 C(=O)(C1SCCc2ccccc21)N1CCN(C(c2cnc(C)o2)=O)C(C)C1C c1(OC)ccc(Br)c2[nH]c(C(N3CCOCC3)=O)cc12 c1(OC)ccc(NC(=O)C(=O)NC2CC(C(F)(F)F)C2)cc1NC(C)C c1(OC)cccc(Cl)c1C(=O)NCC1(CNC(c2c(C)cccc2O)=O)CC1 C1(CNC(CN(C)C)=O)CN(C(C2(C)CC(C3CC3)=NO2)=O)CC12CCC2 CCC(C(=O)NCCCN(C(=O)CN(C)C(C)C)C(C)C)S(N)(=O)=O.C(N)(=O)N c1(C(N2CCN(Cc3csc(Br)c3)CC2)=O)cccn(C2CCSC2)c1=O C1(NC(C(CC(F)F)N(C(c2c(CC)nc(C)o2)=O)C)=O)CCN(C)CC1(C)C C1(NC(=O)NC(C(N2CC(COCC)C2)=O)C)CC1C1CC1 N1(C(C(C(=O)OCC)F)=O)CC2CC1CN(C(=O)CC13CC(C1)C3)C2 N1(C(C2C(C(C)C)OCC2)=O)CCC2CN(C(c3cccc4c3CCC4)=O)C2C1 CCCC(C(=O)N1CC2CCC(CNC(=O)C(CCC)NC(N)=O)C2C1)C(C)C C(C(C)(O)CC(=O)N1CCN(C(c2ccccc2OC)=O)C(C2CCC2)C1)OC C1(CCC(N)=O)CCN(C(=O)CC(=O)OCC(F)F)C1 c1(C(N(C(C)C(=O)NCCCNC2CCCC2)C(C)C)=O)nccnc1N N1(C(C(CC)(C)C#N)=O)CCC(C(=O)N(CCCCO)C)CC1(C)C c1(CC(=O)NCC2CC2N(C(=O)CC2CCCCC2)CCO)cccc2c1OCO2 Cc1cc(C(=O)N(C)CC2CCN(C(c3ccns3)=O)C2)cc2c1CCC2 C1(C(=O)Nc2ccnn2CC(F)(F)F)CCN(C(c2cccc(Br)n2)=O)CC1O c1(C(=O)NCCCN2CCC2)cn2cc(Br)sc2n1.CCOC c1(C(=O)NCCCCCNC(C(C)SC)=O)cc2c(Cl)cccc2s1 C(=O)(CCCCCC(C)C)NCCN1CCCN(C(Cc2c(C)nc(S)s2)=O)CC1 C=C(Cl)CC(C(=O)N1CCCCC1CC(N)=O)NC(=O)C=CC1CCCC1 CN1CCN(C2CCN(Cc3sc(I)nc3Cl)CC2)CC1 N1(C(C=CCOC)=O)CCN(C(=O)Cc2ccc(OC)cc2)C(C)C1C C(=O)(C1=C(C#N)CCC1)N1CC(O)CC(NC(c2cccc(SC)c2)=O)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCCCC(N(C)C(c2cc(CC)no2)=O)C1 c1(C(N2CCCC(C(C(=O)NCc3c(C)scc3)C)C2)=O)cnc2n1CCC2 c1(C(=O)OCC)cc(S(=O)(=O)NCC(C)(O)CC(C)C)ccc1C N1(C(C2C(C#C)C2)=O)CCC2(CC1)CCN(C(=O)CSc1cc(C)cc(C)c1)C2 C1(NC(=O)C=CCN2CCCC2)CN(C(C2CC2F)=O)C2(CCCC2)C1 N1(C(=O)CCc2cnc[nH]2)CCC2(CCCN(C(c3cc(F)cnc3Br)=O)C2)C1 C1(CC(N)=O)(NC(CC2C(C)CC2)=O)CCN(C(=O)C=C2CCC2)CC1 c1(C(N2CCC(F)(F)C(NCc3csc([N+](=O)[O-])c3)C2)=O)ccc2n[nH]cc2c1 C1(C(N2CCOC(CCNC(=O)C(F)(F)C3CC3)C2)=O)COCC2(CCC2)O1 CCC(O)CC(=O)N1C(C(N2CCOC(C(N)=O)C2)=O)CC2CC12 C1(S(N)(=O)=O)(N(C)CCNC(C2(C3CC3)CC2)=O)CC1.c1(C)cn(CCOO)nn1.NCC CC(CC=Cc1ccccc1)C(=O)NCC1(CNC(=O)CN2CCCCC2)CC1 c1(NCC(C)Cn2cccn2)ccc(S(=O)(=O)NCC(CO)C2CCC2)cc1Cl N1(Cc2cc(C)c(Br)cc2)CC2CC(CN(C(=O)C(C)(C)CCl)C2)C1 c1(C(=O)NCCN(C(C)C)C(c2ccoc2Cl)=O)noc2c1CCCC2 C(N=c1nc(N2CCCC3(C2)CC3(F)F)c2c([nH]1)c(C)nn2C)c1cc(C)on1 C1(NC(c2c(OC)n(C)nc2)=O)CCC(C)N(C(C2CCC(C)(O)CC2)=O)C1 Cn1c(O)nc(NCC2CN(C(c3cc(F)cc(F)c3)=O)CCCO2)cc1=O c1(NC(C2CC3CC3N2Cc2cccc(F)n2)=O)ccc(F)c(Cl)c1F N1(C(C2(CNCCOCC)CC2)=O)CCC2(CC1)CC(C(F)(F)F)CO2 C1(NC(C2C(C)COCC2)=O)CC2CCC1N(C(=O)CSc1nccn1C)C2 c1(NC2CCCC(C(=O)Nc3cc(OC)nc(C)n3)C2)ncc2c(ccn2C)n1 c1(C(=O)NCCC(C)(C)NC(c2n(CC)ccn2)=O)cc2c(Br)cccn2n1 c1(OC(C)C)ccc(C(N2CCC23CN(C(=O)OC(C)(C)C)C3)=O)c(C#N)c1.C(Cl)O N1(C(CNC(=O)OCC)=O)CC(O)(CNC(c2cc[nH]c2C)=O)C1 c1(CCCC(=O)NC(C(C)C)C(C)NC(=O)Cn2ncnn2)cc(F)ccc1F C(=O)(CCCC(=O)N(C)C)N1CC(CNC(CCOCCOCC)=O)OCC1 N1(C(C#CC(C)C)=O)CCC2(CCCC2NC(=O)Cc2cc(F)c(N)cc2F)C1 C1(CNC(C(C(CC)O)C)=O)CCN(C(=O)Cn2ncc(C)c2N)CCC1(F)F n1(CCC(=O)N(CC(CC)NC(=O)Cn2ncn(C)c2=O)CC)nc(C)nc1C S(=O)(=O)(c1c(Cl)cccc1Cl)N1C2C(C(=O)NCc3cc(Cl)ncc3F)C(C2)C1 C1(C(=O)NCC(CC)NC(=O)CC2(COC)CCSCC2)CCN2CCC1C2 C(=O)(C(=O)NNC(=O)CSc1ccc2c(c1)CCCC2)OC Cc1cc(=NC(=O)C(=O)NC(C)C(CO)NC(=O)C(O)CCC(C)C)[nH]o1 N1(CC)C(=S)NC(c2ccc(OC)c(OC)c2)C(C(=O)OC)=C1C(F)Cl c1(C(=O)NCC2N(C(C3C(C)C3)=O)CC(O)C2)nc(Br)cnc1N C1(C(N2CC(NC(CN3CC(C)(OC)C3)=O)C(O)C2)=O)CCC2CC2CC1 c1(C(=O)NCC2OCCC(NC(=O)Cc3ccon3)C2)ccc(Cl)c2occc12 C1(CC(=O)NCCC2(NC(CN(C3CCSC3)C)=O)CCC2)COCCOCC1 C1(NC(CCCCC)=O)CCCC12CN(C(=O)C(c1ccc(OC)cc1)C)C2 C1(NC(C(C(C)C)SCC)=O)CCCCN(C(c2cc(N)cc(F)c2)=O)C1 C(=O)(CCCC(C)(C)NC(C1CCCSC1)=O)N(C1C(C)COCC1)C c1(C(=O)NCC(c2cccnc2)NC(=O)CO)cnn2cccnc12 N1(C(c2c(C)ccc(C)n2)=O)CCCC2C(CCCN2C(c2ccn(C)c2)=O)C1 C12(CC(N3CCC(C)(CNC(C4CCCS4)=O)C3)=O)CCC(CC1)OC2 C(=O)(C1=CC(C)(C)C1)N(C(C)CN(C(=O)Cc1nncn1C)C)C C1(CCNC(C2C(CNC(C3(C=C)CCC3)=O)C2(C)C)=O)CCOC1(C)C c1(C(CNC(C(n2cc(CC3CCCCO3)nn2)C)=O)=O)cc(F)cc2[nH]ncc12 Cc1cc(N)cnc1C(=O)N(C(C)C(N1CCC(NC(N)=O)C1)=O)C1CC1 C1(NC(C(CC(C)C)OC)=O)CCC2(CC1)CN(C(=O)CCC(C)OC)CCO2 C(=O)(CS(=O)(=O)C(C)C)NCC(c1ccc(F)cc1F)NC(CNC(=O)OC)=O Cc1c(C(=O)N(C)CCN(C(=O)C(F)=CCCF)C)ccc2ccccc12 CCCC(CNC(C)=O)C(=O)NC1C2CC1N(C(c1ccsc1OC)=O)C2 N1(C(C(c2n(C)cnc2)O)=O)CCC(C2CC2)(CNC(=O)COCCF)C1 C(=O)(C1=CC2CCCC12)NC1(C2CN(C(c3c(N)cc(F)cc3)=O)C2)CC1 N1(C(C(C(C)NC(=O)C=CCO)C)=O)CC2(CCC(C)OC2)C1 n1(C(C)C)cnc(C(=O)NCC=CCC(=O)NCC2CCCCO2)c1 CC1(C)CC(C(=O)NC2COC3(C2)CN(C(=O)CC2=CCCC2)C3)CC(C)(C)O1 C(=O)(C(O)C(F)(F)F)NCC(C(=O)NCCc1ccn(C)n1)OC c1(CNC(c2nnnn2C2COC2)(CNC(=O)OC)C)cc(Cl)c(C)cc1Br c1(CNC(c2ccc(Cl)o2)=O)nocc1C(=O)NC1CCOC1C1CC1 N1(C(C(COCC)N=[N+]=[N-])=O)CCC(C)N(C(=O)CCC(=O)OC)CC1 Cc1noc2cc(C(=O)NCC3CCCC3C(=O)O)ccc12 c1(NC(=O)NCCNC(c2cccs2)=O)cc(C(F)F)ccc1O c1(CC(=O)N(C)CCOCC(=O)NCCC2(C(C)(F)F)CC2)ccnc(O)c1 c1(C(N2C(CNC(CSC)=O)CCC(C)C2)=O)cccn2nnnc12 Cn1cc(C#N)cc1C(=O)NCc1ccsc1C(N1CC2(CC2)C1)=O C1(CC)CCN(C(C2CCC(CNC(C3(C)CCCCC3C)=O)O2)=O)CCO1 Cc1c(C(N)=O)cccc1C(N1CCC(C(C)(C)CNC(=O)COCCF)C1)=O Cc1nnc2n1C(C(=O)NC1CC(N(C)C(c3cccc[n+]3[O-])=O)C1)CC2 N1(C(Cn2c(C)ccn2)=O)CCN(C(C2CCC(C)CC2)=O)C(C)CC1C C1(CC)CN(C(c2sccc2C#N)=O)CCC1NC(=O)Cc1ccsc1Cl C1(C)(NC(C2CC(CC)C2)=O)CCN(C(=O)C=CCn2cncn2)C1 n1(CC(N2CC(C)C(NC(C3(O)CCC3)=O)C2)=O)ccc(O)nc1=O Cc1ccc(C)c(OCC(=O)N(C)CC2(C)CCCC2NC(c2csnn2)=O)c1 C1(CNC(c2cnc(OCC)nc2)=O)CCN(C(=O)CCc2ccco2)CC1C Cc1cccc2[nH]cc(C(=O)NC3CC4CC(NC(=O)CCC(C)(F)F)CC34)c12 N(C1CN(C(C2CN(C)C2)=O)CCc2ccccc21)C(Cc1c(C)nc(S)s1)=O CN1CCN(C(c2cnc(S)nc2)=O)C(CNC(C23CC(F)C2C3)=O)C1 C(=O)(C(C)(CC)C(N)=O)NCCC1N(C(c2ccc(CC)c(N)c2)=O)CCCC1 c1(CC)c[nH]nc1C(=O)NC(C)C(C)NC(=O)Cc1csnc1C CCC(C)C(O)CC(=O)NC(C)CCC(N1CC(C#N)C2(CC2)C1)=O C1(CNC(C2(CC)CCC2)=O)CC(C)(C)CCC1NC(c1cnc(O)cc1C)=O C1(C(=O)NCCCCCNC(=O)CSc2nncn2C2CC2)CCCCC1O C1(F)(CCNC(=O)NC(C2(C)CC2(F)F)=O)CC(NC(C2(C(C)(C)C)CCC2)=O)C1 Cn1c(C(=O)NCC(CNC(C2CC23CC3)=O)CO)cc2sccc12 c1(NC(N(C)Cc2ccc(OC)cc2OC)=O)ccc2c(c1)C(C)(C)CCC2 Cc1nc(C2CC2)oc1C(=O)NCC(C)(O)CNC(C1(C(F)F)CCCCC1)=O C(=O)(CCCN=[N+]=[N-])NC1C(NC(C(=Cc2ccncc2)C)=O)CCC1 CC1(NC(c2cc(C(F)F)cs2)=O)CCN(C(C2CCCC(=O)O2)=O)C1 N=c1ccc(C(N2CCCC(CNC(=O)CC3CC(=O)NC3=O)C2)=O)c[nH]1 c1(C(=O)NC2(C)CC(NC(C(C(C)C)n3cnnn3)=O)C2)cncc2nc[nH]c12 C(N=c1ccnc[nH]1)C1N(C(c2ccnc(Cl)c2)=O)CCOC1 C1(C(=O)NCC(C)(C)OCC(=O)NCC(C)(O)CO)(CO)CCCCO1 c12cc(ns1)C(=O)N(C)CCCCNC2=O.C1(C)(CC)CCCOC1 c1(NC)cncc(C(=O)NCCNC(=O)C(F)OC)c1 C1(C(N2CCCCC(CNC(=O)C(F)CC3CC3)C2)=O)CCc2nc(O)[nH]c2C1 S(=O)(=O)(c1cccc(=NCCO)[nH]1)N(C)C(C)C.C(C)(C)(CC)CC(=C)Br CC(O)CCCNC(C1CCC(NC(=O)Cc2ccccc2)C1)=O C1(C(=O)NCc2cnc(C)o2)(CNC(=O)CC2CCC3CC23)CC(C)(C)C1 c1(C(=O)NCCC(CNC(c2c(C)nncc2)=O)O)cnc2c(C#N)cnn2c1 c1(C(N2CCN(C(C(C(=O)NC)(C)C)=O)CC2C)=O)cccc2cccnc12 CC(CCc1nc(-c2cncn2CC(=O)O)no1)CC(C)(C)C CC1(C)CC(NC(=O)C=CC2CCCO2)CN(C(=O)CC2CCCC2O)C1 c1(CCN(C)NC(C(C)OCCOC)=O)cn(C2C=CCCC2)nn1 C1(CC(=O)N(CCN=[N+]=[N-])C)CCN(C(=O)C(F)(F)C2CC2)C1.C12CCCN1C2 C=C(C)CCCC(=O)N1CCCCCC1.C1(C)C(=O)NCCN1C N1(C(c2ccc(C(=O)NC)nc2)=O)CCCCC(N(C(=O)CSC(F)F)C)C1 C1(C(=O)NC2C(C)N(C(c3coc(C(N)=O)c3)=O)CC2)CCc2n[nH]cc2C1 N1(C(C(F)=CCC)=O)CCC2CCN(C(c3cc(F)c(F)cc3OC)=O)CC12 C(c1cncnc1O)=CC(=O)NC(CCCNC(c1c(OC)nn(C)c1)=O)C Cc1ccc(F)c(C(=O)NC2CC2CNC(c2ccc(N)cc2F)=O)n1 c1(OC)cc(C(=O)NCC(CC(C)C)NC(C2SCCCS2)=O)nnc1C1CC1 C1(CNC(C2(C)CCOC2)=O)CC12CCN(C(c1ccc(Cl)cc1N)=O)CC2 C1(CC)CN(C(=O)CN(C)C)CC1(C)C.c12ccc(cc1)CCC(=O)NC2=O N1(C(=O)NC(CC)CN2CCCC2)CCC(Oc2ccccc2C)CC1 C1(NC(C2(CC(C)C)CC2)=O)CCN(C(=O)CC(C)N2CCCC2=O)C1 CC1(C)CCC(C)(C(N2CCCCC2CNC(C2CCC3CC3CC2)=O)=O)CC1 c1(C(N2C(CNC(C3(N(C)C)CC3)=O)CC(OC)C2)=O)ccc(F)c(Cl)c1N CC1C=C(C(=O)N(C2CCCCN(C(c3ncoc3-c3ccon3)=O)C2)C)CC1 Cc1c(C(N2CCCC2C(N2CCC3(CCCC3)C2)=O)=O)cccc1C#N C(=O)(C1Cc2ccc(Cl)cc21)N1CCCC(C)(C)C1CNC(C1CCCC1)=O C#CCCC(O)C(=O)NCC(C)(O)CNC(=O)C=CCN1CCC1 C12(C(N(C)CC3N(C(C=CCOC)=O)CCOC3)=O)CCCN1S(=O)(=O)CC2 N1(C(CCCC(OC)OC)=O)CC2(C1)C(NC(C1CCC1)=O)CCS2(=O)=O c1cc2cc(c1)-c1cn(nn1)CN2C1CCCCC1.C1(OCC2CC2)CCCC1 Cc1nc(C(=O)NCC2CC2NC(=O)Cn2ccnc2C(C)C)ccc1[N+](=O)[O-] C(=O)(C(O)CC(C)(C)C)NCC1(O)CC(C(=O)NCc2c(C)cccn2)C1 c1(CNC(C2CCN(C(c3ccco3)=O)CC2)=O)c[nH]nc1C1=CCCCC1 C1(C(N2CCC(N(C)C)C2)=O)(CNC(=O)COC2CC(CCF)C2)CCCC1 C1(NC(Cc2c(C)nc[nH]2)=O)CCN(C(=O)C(N2CCSCC2)C)C1C c1(-c2ccc(C(C)=O)cc2F)cc(C(C)(C)C)cc2c1OCO2 C(=O)(C1c2ccccc2OCC1(C)C)NC1CC(NC(CCOCC)=O)C(O)C1 C(=O)(C(F)(F)CCn1cc(-c2nccc(OC)n2)nn1)N1CC=C(C)CC1 C1(C(N(CCCNC(C2CCCCO2)=O)CC)=O)COc2c(F)cc(F)cc2C1 C1(CN(C(C2CC(=O)N(O)C2)=O)CC)CCCN(C(c2cc[n+]([O-])cc2)=O)C1 c1(C(N(C2CCCN(C(CNC(CC)=O)=O)C2)CC)=O)ccc(OC)nc1C C(=O)(C1=C(C)S(=O)(=O)CC1)NC1CN(C(C2(CCC)CC2)=O)CC(O)C1 C12(C(N3CCC3CNC(C(C)OC(CC)C)=O)=O)CCCN(CC1)C2 CC1C(C(=O)NC2(C)CCCCC2C(=O)NCC2CC2(Cl)Cl)=NOC1C Cc1nc(SCC(=O)NCC2CCC3CC2C3(C)C)c(C(N)=O)c(C)c1C CC1CN(C(C23CCC(CC2)C(C)(C)O3)=O)CC2(CCN(C(=O)C(C)C#N)C2)O1 c1(OCC)ccncc1C(=O)NCC1CCCN1C(=O)C=Cc1ncc(C)[nH]1 c1(C(=O)NCC2CN(C(Cc3cc(C)[nH]n3)=O)C(C)(C)C2)nc[nH]c2nccc1-2 C(=O)(C(C)CCC(C)(C)C)N1CC(C)(NC(C(C)C2(O)CCC2)=O)C1 c1(-c2onc(N)n2)cccc(F)c1.n1(CCNC(=O)NC2CC(C)C2)cncn1 C(C(C(=O)N1CC(N(C(=O)C(C)OCCN(C)C)C)C1)OC)OC.C1CC1 N1(CC)CC(NC(=O)CC2CCN(C(C34CC(CN3C(C)C)C4)=O)CC2)CC1=O c1(C(=O)NC2C3(CC(NC(c4cnns4)=O)C3)C2)c(F)ccc2ccoc12 CC1(C(N2CCC(NC(C3CC(O)C3)=O)CC2)=O)CCCC1(F)F C1(N(C(Cc2nc(C)oc2)=O)C)CN(C(C2CC(O)CN2C(N)=O)=O)CCC1C C(N=c1nc(C2CC2)[nH]s1)C1CN(C(C(Cc2cnc[nH]2)NC(C)=O)=O)CC1C N1(C(C=NOC)=O)CC(NC(=O)Cc2ccnc(O)c2)C(CC)C1 N1(C(CCC(=O)OC)=O)CCOCC(F)(CNC(=O)Cc2cccs2)C1 Cc1cccc(C(=O)NC2(C(N3CC4(CC4)C3)=O)CCCC2C)c1C c1(C(N2CC(C)C(C(=O)NCC(F)Cl)C2)=O)ccc(N)c(F)n1 c1(C(N(CC(C)N(C(COC)=O)C)C)=O)csc2cc(Cl)cnc12 c1(C(C)C(=O)NC(C)(CNC(C2(c3cc[nH]n3)CC2)=O)CO)ccc(Cl)cc1 N1(C(CC(CNC(CNC(CCC)=O)=O)O)=O)CCC2(CCC(OC)C2)C1 Cn1cc(S(N)(=O)=O)cc1CC(=O)N(CC1=CCSC1)C C(=O)(C1=CC2CCCC12)N(CC(CNC(c1ccc(OC)c(O)c1)=O)(C)C)C C(=O)(CCCCCN(C)C(C1CC2C=CC1C2)=O)N(C)CCOCCO N1(C(C(C=C)(C)O)=O)CCC(O)(C2(NC(c3cnc(CC)nc3C)=O)CC2)CC1 c1(CN2CC(C(=O)Nc3ccc(C#N)s3)C2)ccc(F)nc1F C=CCC(CC=C)C(=O)NC(CCSC)C(=O)NCC1(C2CC2)CC1 c1(N2CC(=C(CNC(CCCC(C)C)=O)F)C2)ccc([N+](=O)[O-])cc1Cl C1(CC(=O)NC(c2cnn(C)c2)C)CC(F)CN1C(=O)CCC(C)N(C)C c1(CC(=O)NC(C)CN(C)C(C2C=CCCC2)=O)ccnc(O)c1Br c1(C(=O)NCC2N(C(COCCC)=O)CCC2)ccc2nc(Cl)ccc2c1 C12(CNC(c3cc(CC)n(CC(=O)O)n3)=O)CC1CCCN2C(C)=O C(=O)(C1=Cc2ccccc2C1)NCCC(=C)CNC(c1ccc(Cl)c(OC)c1F)=O c1(CC(N2CCCCC(NC(c3[nH]n(C)c(=O)n3)=O)C2)=O)cnn2ccccc12 c1(-c2c(C#C)cccc2)nnc2n1CCCC2c1nc(OC)ns1 C12(CNC(CC(CC)C)=O)CC(NC(C3CC4OC3C3CC43)=O)(CCO1)C2 c1(C(=O)NCCCN(C(=O)COC(F)F)C(C)C)cnc2ccc(C#N)cn12 N1(C(CCOc2ccc(C)cc2)=O)CC2(CC(NC(=O)Cn3ccnn3)C2)C1 c1(C(=O)NC2CN(C(C(C)OCC=C)=O)C2)ncn2c1COCC2 C(CNC(=O)Cn1cnc(C#N)n1)(CC(=O)NCC1NC(=O)NC1=O)OC C=CCC(C(=O)NCC(CC(C)C)NC(c1ncc(OC)cn1)=O)NC(C)=O Cc1nsc(C(=O)NC2(CO)CCN(C(C3CC(N(C)C)C3)=O)C2)c1N N1(C(C(CCOC)C)=O)CC2(C1)OC1(C)CC2(NC(C2CCCC2(C)C)=O)C1 c1(CCC(=O)Nc2c(C(=O)OC)nccn2)cccc(SC)c1O.C12CCN1C2 c1(CN(C(CCNC(c2cnn(C)c2)C)=O)C)ccc([N+](=O)[O-])cc1Cl c1(C(=O)NCC(CN(C(c2cnc(C)s2)=O)C)O)ccc(-c2cccs2)cn1 N1(C(C2CN(C(N)=O)C2)=O)CCC(O)CC1C(=O)NCc1nnc(O)o1 N1(C(c2n(CC=C)ccc2)=O)CCN(C(=O)C=COCC)C(C(C)C)C1 C12(C(=O)NCC(C3CC3)NC(C3CSC3)=O)CCCCC(F)(C1)C2 N1(C(=O)NC(C)CC(N)=O)CCCC(C2CCN(C(=O)Nc3ccccc3)C2)C1 c1(C(=O)NC2(CCCNC(c3cc(CC)nn3C)=O)CC2)cnn2ccncc12 Cc1ccc(-n2nc(CC3CCC3)nc2CN2C(C)CCC2C)cc1Cl N1(C(Cc2cnn(C)n2)=O)CC(NC(=O)CCOCC(F)(F)F)C(C(F)F)C1 c1(-c2scc(CC(=O)NCC(CNC(C(C)SC)=O)C)n2)cccc(Cl)c1 N1(C(=O)NC(c2ccccc2)C(C)C)CCCC1CCC(=O)N1CCCC1 C1(CNC(C=CC(=O)OCC)=O)CN(C(=O)CC2C(=O)NN=C2C)CC1OCC CC(C)CC(C)(O)C(=O)NCCCCc1cn(-c2cnccc2Cl)nn1 C1(NC(C(C)OC)=O)CN(C(c2csc(C)c2)=O)CC2(CCC2)C1 Cn1nnc2cc(CNC3CC(NC(C4CCC(C)(O)CC4)=O)C3)ccc12 c1(CC(=O)NC2(CNCc3ccc(C(=O)O)cc3)COC2)ccc(Cl)cc1F c1(OC)cccc(NC2CN(C(=O)C3=CCC3)CC2(C)C)c1[N+](=O)[O-] C1(NC(=O)CSc2ccncc2)CCN(C(C2CCCSC2)=O)CC1CO c1(Cn2cc(CCN(C3CCNC3=O)C)nn2)ccccc1C(=O)N(C)C C1(C(N2CC(F)(CNC(c3c(COC)ccs3)=O)C2)=O)CCCNC1=O C1(CNC(C(C)CC2CCCCC2)=O)CN(C(C2(F)CCCC2)=O)CC12CC2 N1(C(=O)CCC2CC2)CC(O)CC1CC1CC1.N12CCCC(C1)Cc1cn2nn1 Cc1ccc(F)[nH]c1=NC(=O)c1nccc2c1CCCC2 CCCCC(CN=c1nc(Oc2ccccc2)cc(CC)[nH]1)NC(=O)C#CC c1(-n2c(-c3ccn(C)n3)nc(CC(CC)C)n2)ccc(OC)c(OC)c1 O=C(C1=CC2C=CC1C2)N1CC(C(N2CCCC23CCOC3)=O)C2(CCC2)C1 C1(CN(C(c2cc(CC)[nH]n2)=O)C)CN(C(C2CN(C)CCO2)=O)CCO1 c1(OC(c2ccc(CC)s2)=O)ccc(Nc2ccc(C(N)=O)cc2)cc1F C1(NC(CC2(COC)CCCC2)=O)CCC2CCN(C(C3CCC=CO3)=O)C1C2 CC1C(O)CCCN1C(c1ccc(NS(=O)(=O)Cc2ccc(Cl)cc2)cc1)=O N1(C(C2CC(C)NC(=O)C2)=O)CCOc2ccc(Br)cc2C1 N1(C(C2(N(C)C(C3(CCCF)CC3)=O)CC2)=O)CCC2(CC1)CSC2 C1(N(C(C(=CC2CCCC2)C)=O)C)CN(C(=O)CCCCn2ccnn2)CC1F N1(C(C2C(C)(CC)C2)=O)CCN(C(c2cc3n(n2)CCO3)=O)C(C2CC2)C1 C1(C(=O)O)CCC(C(=O)Nc2ncccc2Cl)CC1 c1(C2CN2C)ccccc1.C1(CO)CCN(C(=O)NC(=O)CCn2cnnn2)C1 C(=O)(CCCCCNC(=O)C=Cc1ccncn1)NC(c1cccc(F)c1)(C)C C(CCC(=O)NC(CCOCC(=O)NC(C)C)c1cn[nH]c1)OC(CCC)=O c1(CC(=O)NCC(CNC(C=C(COC)C)=O)C)c[nH]c(=N)nc1O C(C)(CC(C)CC(C)C)(c1nnnn1C(C)(C)CC)NC(C1(SCC)CC1)=O C(=O)(CC1=CCN(C(=O)C#CC(C)(C)C)CC1)N(C)Cc1ccncc1 C(CC(=O)N1CC(O)(CCNC(=O)C(C)OCC)C1)(C(C)C)OCC c1(OC)c(C(=O)N(C2CN(C(=O)CSC3CC3)CC2O)C)cccc1[N+](=O)[O-] C(=O)(C(O)CC(C)C)N1CC(C(N2CCC2(C)C(C)C)=O)(SC)C1 CCCC(C(=O)NCCC1(NC(=O)CCCn2nc(C)cc2C)CCC1)N(C)C N1(C(C=CCCC)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)CC Cc1nc(C(C)C)oc1C(=O)NCCC1(O)CN(C(=O)Cc2csnn2)C1 c1(C(=O)NCC23N(C(C4(C(C)C)CC4)=O)CC(CC2)C3)onc2ccccc12 c1(C(=O)NCC2(C(=O)NCC(C)(C3CC3)OC)CC(C)(C)C2)nc(C)ccc1C c1(C(N2CC(CNC(C(C)C3CC3)=O)C(O)C2)=O)ccc2ncccc2c1Cl c1(NC(CCNC(C(CC(C)C)N(C(=O)OCC)C)=O)=O)ccc(O)c(=O)cc1 c1(NC2CC3(CC(NC(C(C)OCC4CC4)=O)C3)C2)cc(=O)n(C)c(O)n1 N1(C(C(c2cnn(C)c2)OC)=O)CC(CNC(C2CCC(C(N)=O)O2)=O)(OC)C1 N1(C(c2scc(COC)c2)=O)CCC2C(CCCN2C(C2C3CC4C(C3)C24)=O)C1 C(C)(CCC(=O)NC1(CNC(c2cc(C3(C)CC3)on2)=O)CC1)NC(C)=O c1(C(N2CC(O)(COC)C2)=O)ccccc1-n1cc(C2(C3CC3)CC2)nn1 CC(C)CC(C(=O)Oc1cccc(NC(CC(=O)O)C(F)F)c1)C(C)C C(=O)(CC1OCCc2ccsc21)NCC(C)N(C)C(c1csc(Cl)c1)=O N1(C(Cc2nc(C)[nH]n2)=O)CCCC(C)(CNC(C2CC3OC2C2CC32)=O)C1 C=CCC(CNC(c1cc(C)sn1)=O)C(=O)NCC(N1CCCCC1)C c1(C(=O)NC23CCN(C(CCCOC)=O)CC2C3)cc2c(s1)CCSC2 c1(C(N2CC(O)CC(NC(CCc3cc(C)[nH]n3)=O)C2)=O)cc2cccn2cn1 c1(N(C)Cc2cccn2C)nc(=NCc2n[nH]c(=N)s2)[nH]c2c(F)cccc12 C(CC1=CCN(C(=O)CNC=O)CC1)NC(CCN(CC)Cc1ccncc1)=O N1(C(C(COC)C)=O)C2CC=C(C(=O)N3CCn4nccc43)C1CC2 N1(C(C=CC2CCN(C(C(CCCC)OC)=O)CC2)=O)C2CCC1CN(C)CC2 CCC(C(=O)NCC(C1CCCC1)NC(C1CC(NC)C1)=O)NS(C)(=O)=O c1(C(N(C2CCCC(NC(C3(F)CCOC3)=O)C2)C)=O)nccn2nccc12 CC(C)CC(F)(F)C(=O)N1CCCCC1CNC(=O)CCOC1CCCOC1 Fc1ccc(CC(C2CCCC2)NCCCn2ccnc2)cc1 N1(C(c2c(CNC(c3cc(C)oc3)=O)ccs2)=O)CC2CCCCC2C1C C1(C(N2CCC(C(=O)OCC)C2)=O)CN(CC2C=CCC2)CC1(C)C N1(C(=O)Cn2ccc(O)nc2=O)CC2(C1)CN(C(C1CC(F)C(=O)N1)=O)CCO2 c1(OCC)c(Br)ccc(C)c1NC(c1cccc(OCC(=O)OC)c1)=O CC1CCN(C(c2nc(Br)nn2C)C(=O)NCCCF)CCC1(F)F Cc1c(NC(C)C(C2CCCCC2)NC(=O)CN2CCCCC2=O)ncnc1Cl C1(NC(c2ncc(CC)cn2)=O)CC=C(C(=O)NCC2(C)CCN(C)C2)C1 c1(C(N2C(C(CNC(CN(C(C)=O)C)=O)O)CCCC2)=O)cc(C)c(C)nn1 c1(NC(CCc2nnc(C)n2C)=O)ccc2c(c1)c(C)c(C)n2C c1(C(N2CCC(CNC(COCCCCC)=O)C23CC3)=O)cc(N)c(F)cc1C N1(C(CC2N(C(C(C)CC(F)F)=O)CCC2(C)C)=O)CCc2ncsc2C1 N1(C(C2(C=C)CCC2)=O)CCCC(C)(CNC(c2ccc(=O)n(C(C)C)c2)=O)C1 C1(C(=O)OC)CC12CCC(NC(=O)Nc1cc(Cl)ncc1Cl)CC2 C(=O)(CCCCCN=[N+]=[N-])NCC1(C(=O)NCCC(CCC)O)CCCO1 c1(OC)ccc(Cl)cc1C=CC(=O)N(CC(C)N(C(=O)Cn1cnc(=N)[nH]1)C)C C1(O)(C(N2CCC(N(C(=O)CN3CCCC3=O)CCO)CC2)=O)CC2CCC1C2 C1(NC(=O)CCn2cc(Cl)cn2)CC(NC(c2cc(Cl)ccc2F)=O)C12CCC2 CC(c1ccccc1)=CC(N1CCN(C(=O)COC2CCCNC2=O)CC1)=O C(N=c1[nH]c(=NCCCC(C)(F)F)c2[nH]ccc2[nH]1)c1ccc(N(C)C)s1 C=CC1CCCN1C(=O)CC1CCN1C(=O)Cn1c(C)ccc1C c1(C(C)NC(C2N(C(CCC(C)C)=O)CC(C)C2)=O)cc(F)ccc1F C1(NC(CCCC#C)=O)CCC2CCN(C(C3CC(C)C3)=O)C1C2 C1(c2onc(COC)n2)(C2CC2)COCCN1C(c1cc(O)cc(F)c1)=O N1(C(CCC=C)=O)CCN(C(c2coc(C(F)F)c2)=O)CC2CCCCC12 CCCCC(C)(F)C(=O)NCC.C12CCN(CC1(F)F)C(=O)C(=O)NCC2 C1(NC(=O)CC2(CO)CCCCC2)CCN(c2ncc(O)cn2)CC1O c1(C(N2C(CC)C(C(=O)NCCCOCCO)CC2)=O)cc2n(n1)CCO2 C1(CC)CN(C(=O)C(F)C2CCC2)CCC1NC(c1cnc(C(C)OCC)s1)=O c1(OC)ccccc1SCC(=O)NC(C)C(C)NC(c1ccncc1C)=O c1(Cc2nc(-c3ccc(CCC)o3)n(CC3(C)CC3)n2)cccc2ccccc12 c1(C(=O)NC23CCN(C(C#CC(=O)N(C)C)=O)CC2C3)ccc2ccnc(O)c2n1 N1(c2ncnc(N(C)Cc3c(OC)cccc3)c2C)CCC2(CCC(OC)C2)C1 N1(C(C2CCN(CC)C2)=O)CC(F)(F)CC1CNC(c1cc(SC(F)F)c[nH]1)=O C(C(F)(C(=O)N(C)Cc1occc1C)C(C)C)NC(C1(CC)CCOC1)=O N1(C(c2ncn(CC)c2)=O)C2CCC1CN(C(C13CCCC1(C(N)=O)C3)=O)CC2 C1(NC(C2C(C)(C)C2C#N)=O)CCC(C)(NC(=O)Cc2cc(C3CC3)no2)CC1 N1(C(=O)CCOc2cccnc2)CCC2(C1)CN(C(=O)CSC1CC1)CCO2 C12(OC)CCC(C(=O)NCC3CCN(C(C4(C5CC5)CCCO4)=O)C3)(CC1)C2 C=CC1(C(=O)N(C)CCc2cc[nH]n2)CCN(C(C2CCCCO2)=O)C1 N1(C(CCc2c(C)ncs2)=O)CC(O)(C2CCN(C(C3CS(=O)(=O)C3)=O)CC2)C1 C#CCC(C)C(=O)NCC1CC(NC(c2cn(C(C)(C)C)nc2C)=O)C1 N1(C(C(N2CCC(C)C2)=O)=O)CCC2(CC1)CN(C(C1CCCSC1)=O)C2 C(c1nc2ccccc2s1)=CC(=O)N(C1CC(NC(c2cc(OC)n[nH]2)=O)C1)C c1(CC)cc(C(=O)NCCC2CC(NC(=O)C(C)CN3CCCC3)C2)ncn1 Cc1cccc(C)c1C(=O)NC1CC2(C1)CC(C(=O)NC(C)C(C)(C)O)C2 C1(NC(c2scc(C)c2Cl)=O)CC12CCN(C(C1CCCCNC1=O)=O)CC2 N1(c2nc(C)cc(NC(=O)Nc3cccc(OC)c3)n2)CC(C)OCCC1C c1(OC)ccnc(C(N2CCC(C(C)(C)NC(C34COCC3C4)=O)C2)=O)c1OC c1(OC)c(C(N2CCN(C(=O)C(C)(C)CC(C)C)C3(CC3)C2)=O)cc(F)cc1F c1(-c2nc(CN3CCC(CC4C(=O)OCC4)CC3)on2)cc2ccccc2cn1 C1(CNC(CCOCCSC)=O)CC2(CCN(C(=O)C(C)C)C2)CO1 c1(C(C)C)nn(C)cc1C(=O)NCC1CCCCN1C(C1(C(C)(F)F)CCC1)=O N1(C(C2(C(C)C)CCCC2)=O)CCCCCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C1 Cc1nc2ccc(C(=O)NCCC3CN(C(=O)C=CCF)CC3C)cc2o1 Cc1nn(CC(=O)NCCCN(C(=O)C(C)C(F)F)CC2CCCC2)c(=O)o1 C1(NC(=O)CC23CCCC2C3)C2CCC(C2)C1C(=O)NCc1cccnc1O Cc1nn(C)c2cc(C(=O)N(c3cncc(Br)c3)N3CCOCC3)cnc12 N1(N(c2ccc(NC(C)C)cc2)C(C)=O)CCN(C(=O)OC)C(=O)C1C c1(C(=O)NCC2C(NC(C3CC(C(F)(F)F)(OC)C3)=O)C2)nc2ccccc2o1 n1(CC)nnc(C(N2CCC(C3CCCN3C(=O)CC3OCCCO3)C2)=O)c1C c1(OCCC)ccc(CN(C(c2occc2Br)C(=O)NC2(C)CC2)C)c(C)n1 c1(C(=O)NCC(C(C)C)NC(=O)C(F)C(C)C)cc2[nH]ccc2s1 c1(OCC(=O)NCC2CN(C(CC(CC)C)=O)CC2C)c(C)nn(C)c1C N1(C(CC(C)C2CCCC2)=O)CC(NC(=O)CCc2ccnc(Cl)c2)C(F)C1 C(=O)(C1=C(F)CN(C(c2sccc2F)=O)CC1)NCCCc1nc(C)[nH]n1 c1(C(=O)NCCN(C(=O)CCC(=O)C2CC2)CCOC)ccc2cccnn12 c1(C(N2C(CNC(c3ncc(OC)nc3)=O)C(C)CC2)=O)ccnn2ccnc12 C1(NC(C(C)CSc2ccccc2)=O)(CO)CCCN(C(C2CNC(=O)N2C)=O)C1 CC1CCN(C(c2cccc3sncc23)=O)CCN1c1ncccn1 N1(C(Cn2cnc(C(N)=O)n2)=O)CC2(C1)CC2(F)Br c1(OCCOC)cccc(-c2nc(C(C)OC)n(-c3cnn(C)c3)n2)c1 c1(NC(C2C(NC(C3CCCS3)=O)CCC2)=O)c(Br)cc(F)c(F)c1F Cc1csc2ncc(C(=O)NC(C)(CNC(=O)COCCCF)C(C)C)n12 NC(=O)CC(O)C(=O)NCC1(C(=O)NC2(C3CCCCO3)CC2)CC2(CC2)C1 C(=O)(C(C)(C)CC(F)F)N1CC(C(N2CCC(C=C)CC2)=O)C(CCC)C1 c1(C(C(=O)NCCN(C(=O)COc2cc(Cl)ccn2)C)(F)F)ccc(F)cc1C C1(NC(=O)C(F)CC2CCC2)CC12CCN(C(=O)CCC1CCCCCC1)CC2 C1(NC(c2cc(C)ncc2)=O)CCCCC12CCN(C(=O)CC1CC1C)CC2 c1(SC)ccc(-c2nc(Cc3ccccn3)nn2-c2ccccc2)cc1OC N1(C(c2cc(C)cc(C)n2)=O)CC2CCOC2(CNC(c2cnn(C)c2Cl)=O)C1 Cc1ccc(I)c(NC(C2CC3(CC3)CN2C(=O)CSc2ncccn2)=O)c1 N1(C(c2c(CC)csc2)=O)CCC(C(C)NC(=O)Cc2cncn2C2CC2)CC1 C1(NC(C2C(CCC)C2)=O)(CC)CCCN(C(c2ccnn2CCCC)=O)C1 N1(C(C23CC(C)C2C3)=O)CC(NC(C2(C(=O)NC3CC3)CC2)=O)CC12CCC2 N1(C(C2CC2C)=O)CCC=C(C(=O)NC(c2c(OC)csc2)(C)C)C1 N1(C(c2cc(CC)nn2C)=O)CC2CCCC(CNC(=O)C(F)OC)C2C1 c1(CC(=O)NCC(CC)NC(=O)CC2CCC2(C)C)c(F)cc([N+](=O)[O-])cc1F C(=O)(CCS(C)(=O)=O)N(C)C.C12(C(=O)OC(C)(C)C)CC1CCCN2C=O N1(C(C2CC3(C2)CC(O)C3)=O)CCC2(CCC2)C1.Cn1nc2cc1C(=O)NC2 CC1CCC(CCC(=O)NCc2nocc2C(=O)N(C)CCC2CCCCC2)O1 N1(C(C=CSC)=O)CCC(NC(=O)C=Cc2cc[nH]n2)CC1C CC1(C)CCCc2cc(C(N3CC4CC(Nc5cc(CO)ncn5)C4C3)=O)sc21 C1(C)(C(=O)NCCOCCN(C(CC(C)OC)=O)C)CCC12CCC2 C(CN=C(NCc1ccc(C)cc1)N1CCC(C2CC2)C1)N(C)CCN1CCCC1 N1(C(=O)Cc2ccsc2)CCN(c2ccc(-c3ccc(COC)cn3)cc2)CC1 C1(CCOC)CN(C(C2CCC3CC23)=O)CCN1C(c1ccc(C(F)F)nc1)=O c1(Sc2c(N3C(C)C(=O)N(C)CC3)nccn2)ccc2cccnc2c1 N1(C(C2CN(C3COC3)C2)=O)CCC(C2CCN(C(C3CC(F)(F)C3)=O)C2)CC1 N1(C(C2N(C(C)=O)C(=O)CC2)=O)CC(NC(C2CC2CC(C)C)=O)CC1(C)C c1(CC(=O)NC2CC(OC)CN2C(c2cc(N)ccn2)=O)cnc(Cl)cc1C c1(C(N2C(C(=O)NCc3nccc(C)c3)CCC2C2CC2)=O)cc(C#N)n(C)n1 C1(CCCC)CCCN(C(C23CC2CCN3C(c2nscc2C)=O)=O)C1 CN1C(=O)CSC1=CC(=O)N1CC2CC2(NC(=O)CCNC(=O)C(C)(C)C)C1 C(C)(C(=O)N=c1cc(C)n(C)[nH]1)NC(C(C(CC)C)C(CN1CCCC1)=O)=O N#Cc1ccc(NC(C2CCCCN2C(=O)CCc2ccccc2C#N)=O)cn1 Cc1cc(NC(c2csc(=N)[nH]2)=O)ccc1NC(C12CCC(CO1)C2)=O c1(C(=O)NCC#CCNC(Cn2ncc(C)c2)=O)cccc2c1CCO2 c1(OC)cc(NC(C2(C)CCN(Cc3cccc(C)c3F)C2)=O)ccc1C#N N1(C(C#CCNC(c2cnoc2)=O)=O)CC(F)(F)C1C1CC1 Cc1ccc2[nH]c(C(N3CCC4CCN(C(=O)C(F)F)CC34)=O)c(Cl)c2c1 c1(CC(=O)NC(CNC(c2ccc(C)o2)=O)(C)C(C)C)ccc2c(c1)COCC2 Cc1nc(O)nc(C)c1C(=O)NC1CCCCC1NC(c1ccc(Cl)c(N)c1)=O CCC(C)CC(C)C(=O)NCc1cc(C(N2CCC=C(F)C2)=O)no1 C(=O)(C1=C(C2CCCC2)CN(C(=O)CCC2NC(=O)NC2=O)C1)OC(C)(C)C c1(C(=O)NC2CC(OC)C2)csc(CNC(=O)C(F)C2CCOC2)c1 C(=O)(C(C)CC(F)F)N1C(CNC(c2c(C)n(CCO)nc2)=O)CCCC1 C(=O)(C(C#N)C(C)(C)C)N1C2CCCC2C1.C(CC(=O)NC1CCC1)C1(C)CC1 C1(C(=O)NCCCCCOC)CC(OC)CN1C(=O)CC(C)(C)OC Cn1ncc([N+](=O)[O-])c1NC(C1CCC1CNC(=O)CCCc1cccs1)=O c1(C(C(=O)NC(CC)C)N(C)CCOC)cc(Oc2ccccc2)ncc1Br c1(OC)cnc(C(=O)NCC2CC(O)CN2C(C2CC2C(F)F)=O)nc1 c1(-c2cccc(C(C)O)c2F)cccc2c1CN(C(=O)CS(=O)(=O)CCO)CC2 N1(C(C=CCCC)=O)CCC(C)(C)C1C(=O)NC(C)CN1CCCC1=O N1(C(C(CC(N)=O)O)=O)CC(C2CCCN(C(c3nc[nH]c4nccc3-4)=O)C2)C1 C1(NCc2ccc(C(=O)O)s2)CC2(C1)CC2C(=O)NCCCCC1CC1 CCC(Cc1ccccc1)C(=O)NC1CC(CO)N(C(=O)CCc2cn[nH]c2)C1 c1(C(=O)NCC(CNC(C2(OCC)CCC2)=O)(C)O)ncc(C)cc1OC N1(Cc2cccc(OC)n2)C2CCC1CC(NC(c1cn(C3CC3)nc1C)=O)C2 c1(C(N(C2CCCN(C(=O)C=CCF)CC2)C)=O)c[nH]c2ccc(Cl)cc2c1=O N1(C(c2ccc(COC)cc2)=O)CCCC2(C1)CN(C(=O)C(C)(C)CCC#N)C2 c1(C(=O)OC)ccccc1NC(c1ccc(NC(=O)CSC)cn1)=O c1(CN2CCCC(C)(CNCc3ccc(C=C)cc3)C2)c[nH]c2ncc(Cl)cc12 C1(NC(c2cc3c[nH]nc3s2)=O)CCOC2(CCN(C(C3CCCS3)=O)CC2)C1 C1(NC(C=NOC)=O)CN(C(c2ccc(=O)n(C)c2)=O)C2(CCOC2)C1 c1(OC)cc(NCC2C3CN(c4ncnc5sccc45)CC23)c(Br)cc1Br CC(CN(C)C)CC(=O)NC1(CCNC(c2cc(C3CC(F)(F)C3)[nH]n2)=O)CC1 C1(C(=O)NCC(C)(C)CC2CC2)N(C(=O)CCc2cnn[nH]2)CCCC1(C)C N1(C(c2c(C(=O)OC)csc2)=O)CC(NC(C2(C)CCN(C(C)=O)C2)=O)CCC1C c1(C(=O)NCC2CCN(C(C3(C)CCCNC3=O)=O)C2)cnc2c(F)cccn12 c1(N2CC(OC)C(O)C2)ccc(S(=O)(=O)NCCC=CBr)cc1C#N Cc1cc(-n2cccn2)nc(NCC2CCCN(C(C3CCCOC3)=O)CC2)n1 O=C(C1CCCc2nn[nH]c21)NCC(C1CCOC1)O C(=O)(C(CC(=O)NC(C1CNCCC1C(F)F)=O)C(C)=O)OCC c1(C(=O)NCC)ccc(-c2csc(NC(c3nc(-c4ccco4)n[nH]3)=O)n2)cc1 Cc1onc(C(F)(F)F)c1C(N1CCC(CC(C)NC(c2cccs2)=O)CC1)=O c1(C(N2CCCC(NC(c3sccc3Cl)=O)(CO)C2)=O)cncc2c1CCCC2 c1(C(=O)Nc2ncccc2O)c[nH]c2cc(-c3cc(C4CC4)cnc3F)cnc12 c1(C(=O)NC(C(=O)N(CC#CC)C)Cc2cn[nH]c2)cccc(Cl)c1 C#CC1(NC(c2c(O)nnc(C)c2C)=O)CCC(C)(C)CC1 c1(C(N(CC(C)CNC(c2ccc(-c3ccsc3Cl)s2)=O)C)=O)ccnc(O)c1 Cc1nccc(C(N2C(CNC(=O)C(C)c3ccsc3)CC3CC23)=O)c1O C(=O)(C1COCc2ccccc21)N1CCC(N(C)C(c2cc(Cl)cnn2)=O)CC1 C(=O)(C(CO)C(F)(F)F)N1CC2OCC(NC(CCCCOC)=O)C2C1 c1(C(=O)NC2(C)CC(NC(C3C(C)(C)C3(F)F)=O)C2)cccc2ccnn12 c1(CC)ccc(C(N2CCC(C)(CC(=O)NC3CC(N(C)C)C3)C2)=O)nc1 C1(C(N2CC(=CC)C2)=O)CCCN(C(C2CN(C)CCO2)=O)CC1 c1(OC)cc(F)ccc1C(N1CCCC(c2cc(C)cc(C)c2)C1)=O C=CC1CCCC(NC(=O)C(Cc2cnc[nH]2)NC(=O)CCCCC#N)C1 c1(C(N2CCC(C(c3ccccc3)C)C2)C(=O)NCC=C)csc(C(C)C)n1 C1(C)(CNC(c2cnc(NC)c(Cl)c2)=O)CC(F)(F)CN1C(=O)CCSC C1(C(N2CC(C3(NC(c4c(N)cc(F)cn4)=O)CC3)C2)=O)CCOCC12CCC2 c1(CC(=O)Nc2ccc(C(=O)OC)c(O)c2)cc(F)c(Br)c(F)c1 CP(C)(=O)C1CCC=C1C(=O)NCC1=CCN(C(=O)C#CC2CCOC2)CC1 C(C(CC(C)C)C(=O)N1CCN(C(=O)C=Cc2cccs2)CC1CC(F)F)OC c1(OC)nc(NCCN(C)CCCCO)ncc1Cl.C1(CCO)(C(=O)NC)CC1 C1(C(=O)NC2CC(C)(NC(c3cc(C(C)C)on3)=O)C2)CCOC(C)C1 c1(CN2CC(C(=O)Nc3nc(C)sc3)C2)ccc(N2CCCCC2)cc1 C#CCCS(C)(=O)=NC(=O)c1c(C)nnn1-c1cccc(C)c1 c1(COCCC(=O)NC23CC(NC(CCC=C(C)C)=O)(C2)C3)cccc(Cl)c1 c1(C(=O)NC(CNC(Cc2c(C)non2)=O)C2CC2)cnc(C2CC2)[nH]c1=N c1(C(N2CCC(C)CC2)=O)cc2nccc(C(F)(F)F)n2n1.c12sccc1NC2=O N1(C(c2cc(OCC)n[nH]2)=O)CCC(N(C)C(C2(C)CC3(CCC3)C2)=O)C(C)C1 C(=O)(CCC1=NNC(=O)CC1)NCC1(O)CN(C(c2n(C)cc(C#N)c2)=O)C1 c1(C(N(CCN(C(C2C(=C)CC2)=O)CC)CC)=O)cnc(Cl)s1 N1(C(C(CCSC)O)=O)CCCN(C(=O)CC2CCC(C)CC2)CCC1 CN=c1ccc(C(=O)NC2CCC(CC(=O)N(CCC(=O)NC)CCO)C2)c[nH]1 c1(CCC(N2CC3(CN(C(C4=C(C)CCC4)=O)C3)C2)=O)c(Cl)cccc1[N+](=O)[O-] C#CC1COCCN1C(C1CCCN(C(=O)CC2CCCCCC2)C1CC)=O c1(OC(C)C(=O)NCCCN(C(=O)CC2=CCCCC2)C)ccc2c(c1)CCC2 C(C(=O)N1CCCC1NC(c1ccccc1)C1CCC1)(C(C)C)OC N1(CC(=O)NC23C(CN(C(c4c(C)nnn4C)=O)C2)C3)CCCCCC1=O C1(NC(C2CC(Cl)(Cl)C2)=O)CCC2(CCCN(C(=O)Cc3cncc(O)c3)C2)C1 C1(CN(C)CC2CCN(C(c3nc(C)c(C)s3)=O)CC2)CC2CCC(C1)S2 N1(C(CSc2nc(C)[nH]n2)=O)CC(NC(C2CC(F)C(=O)N2)=O)CC2(CCC2)C1 c1(C(=O)NC(CC)CNC(c2ccc(F)nc2)=O)cn(C)c2c(cnn2C)c1=O C(=O)(CCCCO)NCC(=O)NCC1C(NC(c2cc(C(C)(C)C)[nH]n2)=O)C1 N1(C(C2C(C)(CC)C2)=O)CC(CNC(c2oc(SC)cc2C)=O)CC1C N1(C(N=c2c(C#N)cn(C)[nH]2)=O)C2CCC1CC1(C2)CC1(F)F C(CCC(C)(C)C(=O)NC1CCC1F)NC(CCCC1C(C)C1)=O CCCCC(C(=O)N(CCC#N)CC(=O)OC)N1CCCC1c1cccnc1 C(=O)(CS(=O)(=O)C(C)(C)C)NC(C1CCN(C(C(n2cc(Cl)cn2)C)=O)C1)C C1(C(N2CC(N(C(=O)COCc3ccccn3)C)C2)=O)CC(C2CC2)=NO1 CN(CC(=O)NSS(C)(=O)=O)N1CC2(CCN(C(C)(C)C)CC2)C1 c1(C(=O)NC2CN(C(c3c(C)n[nH]c3C)=O)CC(O)C2)cnc2ccnn2c1 N1(C(C2(C)CC2)=O)CCN(C(=O)CC2SCCS2)C(C2CC2)C1.C(F)(F)F c1(C(C)=O)cc(OC(F)F)ccc1Br.c12cn(nn1)C1(CC1)NC2=O N1(C(c2cc(SC)oc2)=O)CC(CCNC(C2(C)CS(=O)(=O)C2)=O)C(C)C1 C(CCN(CC(=O)NC)C(=O)C(F)(F)C(C)O)NC(CSCC=C)=O N1(C(Cc2cc(C)on2)=O)CCCCC1c1cn(CCC2CC2(Cl)Cl)nn1 C1(C(C)NC(CSCCC)=O)CCCN1C(=O)C(C)COCC C1(C)(C(N(C2CCN(Cc3ccc(C#C)o3)C2)C)=O)CCN(C)CC1 C1(CNC(C(C)N(CCCC)CCC)=O)CC2CCCC2C1.N12CC(C1)C2=O C1(CC(=O)N(CCNC(c2c(CC)ccs2)=O)C)CCC(C)CO1 C1(COC)CCC=CC1NC(=O)CC1CCN1C(=O)CC(C)C1CC1 c1(OC)ccccc1CCC(=O)NC1CC(CNC(C2CC3CCCC23)=O)C1 C1(NC(C2(CNC(c3ncc(C)c(C)c3)=O)CCC2)=O)CC2CC1CC21CC1 c1(C(N2C3CCN(CC3)C(=O)C(O)C2C)=O)cc2c(O)cccc2[nH]1.CC.S(C)C C(CCC(N)=O)(C(=O)N1CC(NC(=O)Cc2cncn2C)C2(CC2)C1)N(C)C C(=O)(CCCCCN(C(=O)Cn1cnc(=N)[nH]1)C)NC(C)Cn1cncn1 C1(NC(C2(C)CCN(C(=O)C=Cc3ccsc3)C2)=O)CCC2CC1C2(C)C C1(COC)CN(C(=O)C(C)N(C(=O)CCC2CCCC2)C2CC2)CCO1 C(=O)(C1=CCC2(COC2)OC1)N1CC(O)(CN(C)C(C2(C)CCCC2O)=O)C1 c1(-c2cc(OC)c(CN(C)C)cc2)cc(C(=O)OC)c(F)cc1NC1CC(O)C1 CC1CN(c2cc(C(C)(C)C)ncn2)CCC1NC(=O)CC1CC1 C1(C(N(CC(CCC)O)C)=O)CN(C)CCN1C(c1cc(C)c(O)nn1)=O C1(CNC(c2n(C=C)nnc2)=O)CN(C(=O)CC2CCC(F)(F)CO2)CCCO1 C(=O)(C(F)(F)CO)NCCC(C)NC(C1CC(OC(F)F)C1)=O CN1CCc2nc(C(=O)NCC3CCCN(C(=O)C=Cc4cnc[nH]4)C3)sc2C1 Cn1nnc2cc(C(N3CCC34CN(C(C3(C#N)CCSCC3)=O)C4)=O)sc12 CCC(CC)CC(C(=O)NC1CC1)N1CCC(F)CC1 C1(NC(C(CC)CC)=O)CC(F)(F)CC1NC(=O)C(C(C)C)NC(=O)OC C(CCC(=O)NC(CCCCO)C(=O)N(C1CC1(C)C)C)OCCOCC N1(C(C(CNC(c2cc(C)on2)=O)C(C)C)=O)CC2CCC1C(O)C2O C12(C(N3CCCN(N4CCC(C=O)C4)CC3)=O)COCC1CN(CCO)C2.CCO Cc1cc(F)c(C(=O)Nc2c[nH]nc2Cl)c(Cl)c1 Cc1ccnc(C)c1NC(C1CN(C(=O)C(C)n2cccc2)CCO1)=O C1(CNC(=O)CCc2nncs2)CCCCN(C(C2CN3CCN2CC3)=O)C1 c1(C(=O)NCC(CC(C)C)NC(C(C)=C2CCC2)=O)cnc(O)c2ccsc12 N1(C(C(C)OCC=C)=O)CCC(NC(=O)CNC(N2CCCC2)=O)CC1C c1(-c2n(C(C)C(F)(F)F)nc(CC(C)(C)CO)n2)cccc2ccn(C)c12 C(=O)(N=c1cnn(C2CCOCC2)[nH]1)N1C(C)(C)CC1 CC12CC(NC(C3CC(=O)N(O)C3)=O)(C1)C1(CN(C(C3CCC(=O)O3)=O)C1)O2 c1(C(N2CCCC(CC)(NC(c3scnc3C)=O)C2)=O)cnn2c1OCC(O)C2 C1(NC(C(c2ccccc2)NC(=O)C(F)F)=O)CCN(CC2CC2)C1 C(CC(O)CC(=O)N(C1CCN(C(=O)CCc2cccs2)CC1)CC1CC1)SC Cc1cc(CC(=O)NC2CC(NC(=O)C(C3CCC(=O)N3)C)C2)ccc1Cl N1(C(c2ccc(CCC)[nH]2)=O)CCN(C(=O)C(=Cc2ccnn2C)F)CC(O)C1 c1(OCC(=O)NCC=CCNC(C(C)N(C(C)=O)C)=O)cccc(O)c1.N C=C1CCN(C(=O)CC(C)(F)F)C(C(=O)NCc2cnc(C)n2C)C1 C1(C(C)(C)OC)CN(C(=O)C(F)=CCCF)CCN1C(=O)CCS(C)=O C#CCC(O)C(=O)NCCN(C(C1(O)CCCCC1)C(=O)NC1CCC1)C C(=O)(C1=CCS(=O)(=O)C1)N(CCCN(C)C)CCNC(=O)C#CC1CC1 c1(C(N2C3(CNC(C(C)(C)CF)=O)CCC3CC2)=O)ccc(S(N)(=O)=O)nc1 CCCC(C)CC(=O)N1CCOC(CC(N2CCCC(OC3CC3)C2)=O)C1 C1(C2CC2)(C(=O)NOCC23COCC2C3)CN(C(=O)C2CC2)C1 Cc1c(C(=O)NC2CCC(NC(=O)C(F)(F)C3CCCC3)CC2)cnn1CCO C1(NC(C=C(C)C2CC2)=O)CCN(C(C2CCCCS2)=O)C1 c1(C(C)(C)C)conc1CNC(c1ccoc1)CO Cc1cnc(C(=O)N(CCCN(C(=O)CCCC2CCCCC2)C)C)c(O)c1 C1(N(C(=O)COC2(F)CC2)CC)CCCN(C(=O)Cc2ccnc(O)c2)C1 c1(CCN=[N+]=[N-])ccc(C(=O)NC2CCOC(C3CC3)C2)cc1 C1(C(=O)NC(CC=CC(=O)NC(c2cc(C)on2)C)(C)C)CC(O)C(F)C1 N1(C(CCC#CC)=O)CCC2(CCN(C(c3ccoc3CC(N)=O)=O)C2)C1 c1(OC)ccnc(CNC(=O)CCNC(=O)CN2CCCC2=O)c1 N1(C(Cc2ccc(C)c(C)c2)=O)CCN2C(CCS2(=O)=O)C1 N1(C(CCc2c(C)noc2C)=O)CC(N(C(=O)COC(C)C)C)C2(CC2)C1 N1(C(C(C(=C)C)(C)O)=O)CC2CCN(C(=O)CN(C)C(C)C)CC2C1 n1(CC)cc([N+](=O)[O-])c(C(N2CCC(NC(c3cc(Br)c[nH]3)=O)C2)=O)n1 Cc1cc(C(=O)NC2COCCN(C(c3ccncc3Cl)=O)C2)nc(C)n1 c1(CN(C)C(=O)NC2(C)CC3(CC3)C2)ccc2c(c1)CCC2 CC1(C)CCC(CNC(c2coc3c2CCCC3)=O)N(C(=O)CCCC2CC2)C1 CCC(CC(F)F)C(=O)N1CCC(C(C)C)CC1CNC(=O)CCn1cccn1 CCCCCC(C)(C)C(=O)N(CC(C)NC(C1OCCC1C(F)(F)F)=O)C C1(NC(CN2C(C)CCC2C)=O)CC2(C1)CN(C(=O)CN1CC=CC1)C2 c1(OC)ncc(C(=O)NC2CCN(C(c3cccc(C)c3O)=O)C2(C)C)c(C)n1 c1(C(=O)NCCCCNC(C2(c3ccc(C)cc3)CC2)=O)cccn2nccc12 Cc1cn2c(n1)CC(C(N1CC3CC1C3NC(=O)Cc1cncs1)=O)CC2 C1(C(C(=O)NC2C(NC(CCN(CC)CC)=O)CC2)NC(C)=O)CCCCC1 C12(CNC(c3c(C)cc(C)s3)=O)CCC1CN(C(=O)C(c1cccnc1)C)C2 c1(C(N(C2CN(C(C3CCC(C(N)=O)CC3)=O)C2)C)=O)ccc(=O)n(CCO)c1 Cc1ccc2nc(C(=O)NC3CC4CC3N(C(=O)C(C)(C)C3CC3)C4)cn2c1 CC1(C)CC(NC(c2csc(Br)n2)=O)CN(C(=O)CN=S(C)(C)=O)C1 N1(C(C2(CC=C)CCCN2C(c2cc(C(C)=O)on2)=O)=O)CC(C2CCCC2)C1 C#CC1CC2CCC1N(c1nc(-c3ccncc3)nn1C)C2 C(CC(CC)C(=O)NCC1(NC(=O)CN2CCCCCC2)CCCCC1C)=CC N1(C(c2c(C)n(C)nc2)=O)CC2(CCN2C(=O)COCC2CCCCO2)C1 Cc1cc(O)c(Cl)cc1C(N1CC(C)CCC1CNC(=O)C#CC(C)(C)C)=O c1(OC)cc(F)cnc1NC(C1(C)CN(Cc2ccncc2)C1)=O c1(C(=O)OC)cc(Cl)c(Cl)cc1S(=O)(=O)NNC(=O)c1onc(Br)c1C Cc1ccn2c(C(=O)N(CC(C)NC(c3scc4c3OCCO4)=O)C)cnc2c1 c1(C(N(C)CC2(NC(c3csnn3)=O)CC2)=O)ncccc1-c1ccccc1 c1(C(COC)NC(=O)CSc2n[nH]c(=N)s2)ccc(F)cc1 c1(C(=O)NCCN(C(=O)CO)CC)coc2c(Cl)cccc12 c1(C(=O)NCC2CCC(NC(CCS(C)(=O)=O)=O)C2)cnc(O)c2cccnc12 Cn1[nH]c(=N)cc1C(N1CC(CO)(NC(=O)CCc2ccccn2)C1)=O CCCCCCC(=O)N(C)CC1CCCN(C(=O)CC(C)n2ccnc2)C1 c1(N2CCCC(CCC(C(CCCC)C)=O)CC2)ncnc2sccc12 Cc1cnn(C)c1C(=O)NC(C)CN(C)C(c1cccc(C(C)C)c1)=O C(=O)(CCCCCNC(C1CC2(CCCO2)C1)=O)NCCCSC C1(NC(CCCCC)=O)CN(C(C2CC(=O)NC2(C)C)=O)C2(CCCCCC2)C1 c1(C(N(C(C)CNC(C2CNc3nccn3C2)=O)C)=O)ccc2ccncc2c1 CC(c1ccco1)=CC(N1C(C(=O)NC2COC(C(C)C)C2)CCC1C1CC1)=O c1(NC2CN(C(C(CC)CO)=O)CC2(C)C)nc(C)nc2[nH]ccc12 Cc1ccc(C=CC(=O)NCC2CC2NC(=O)Cc2c(O)ncnc2O)nc1 CC(C)CC(C)CC(C)C(=O)N1CCCC(N(C)C(C2CCS(=O)CC2)=O)C1 S(=O)(=O)(CCC(=O)NCC(C(C)C(C)C)NC(=O)C=Cc1ncc(C)[nH]1)NC c1(N(CCCOC)C)nnc(N(C2CC2)C)n1Cc1ccccc1 C12CCCN(C1)C(=O)CSCC(=O)N(C)CCOC2.CCC(=O)OCC.N(C)C C1(NC(c2cn(CC)nc2-c2ccccc2)=O)CC2(COCCO2)C1 C1(C)(C(=O)NC(C(CO)NC(c2c(C)occ2)=O)C)CC(F)(F)C1 N1(C(C(COC)(C)OC)=O)CC2CCC(C1)N2C(c1cnn(CCO)c1N)=O C1(NC(c2conc2C2CCC2)=O)CN(C(c2cc[nH]n2)=O)CC2(CC2)C1 C(=O)(CCCCCF)NC(C(=O)NC1(COC)CN(C)C1)c1cccs1 c1(C2(C(=O)NCC=CCNC(C3(F)C(C)C3)=O)CC2(F)F)ccc(Cl)cc1 N1(CCC#C)CCC(C(=O)NCC2CCN2C(=O)CCN2CCCCC2=O)CC1 c1(C(N(C2CN(C(c3ccc(C(=O)NCCO)[nH]3)=O)C2)C)=O)c(C(F)F)cnn1C N#CCS(=O)(=O)c1ccc(C(N2CCCN(C(=O)CC3CC3)CCC2)=O)cc1 Cc1scc(C(=O)NCCC2(C)CCN(C(c3coc(Br)c3)=O)C2)c1C C1(CCOC)CCN(C(=O)C(CCSC)NC(=O)CCCNC(=O)OC)CC1 c1(C(=O)NCC2OCCN(Cc3c(C)nc(CC)o3)C2)cc(C)cnc1F S(=O)(=O)(c1cn(C)cn1)N.C1(CCN(C)C)CCOCC1 C1(C(=O)NC2CC(CNC(C3CN(S(N)(=O)=O)C3)=O)C2)CCc2cnnn2C1 C(=O)(C1CCc2c[nH]nc21)NCCn1cc(C(=O)NCC(C)N=[N+]=[N-])nn1 C(CC(F)(F)F)(C(C)(C)C)C(=O)OC(C)(C)C.C1C(c2ccccc2)C(=O)O1 c1(NC(C2C(CCC)CN(C(=O)C(CC3CC3)OC)C2)=O)ccc(F)c(F)c1 C1(C(N2CC(O)(CNC(Cc3cc(C)on3)=O)C2)=O)COC(=O)N1C C=CCCCCCCC(=O)NCCC1(C)CCN(C(c2cnc(C)s2)=O)C1 C1(N(C(=O)CCCF)CCC)CCN(C(c2cncc(C(=O)OC)c2)=O)CC1 C1(C#N)(C(N2CCC(c3cn(CC(=O)OC)nn3)CC2)=O)CCCCC1 C(C(C)(C)C(=O)NC1CC(C(F)F)C1)NC(C(C)NC=O)=O C(=O)(C(C#N)C(C)(C)C)NCCCCN(C(C1(c2cc(C)no2)CC1)=O)C N1(C(c2cc(C)no2)=O)CCCC(C)(C)C1C(=O)NCCC1CCCC1 N1(C(c2ccc3ncoc3c2)=O)CCC2(CCN(C(c3cnco3)=O)C2)C1 Cc1n[nH]c(C)c1C(C)C(=O)NC(C)CCNC(c1ccc(C(O)CF)cc1)=O N1(C(c2ccc(C)cc2)=O)CC23CCCC2(C1)CN(c1nc(C)ncc1F)C3 c1(C(N2CC(NC(c3[nH]c(C)cc3C)=O)CC(OC)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(NC(C)(C)C)CCOCC12CCCCC2.c12nnnn1NC2CCC1CCC1 C1(C(=O)NCC2CCCN(C(C3CCCCCCC3)=O)C2)CCCCNC1=O n1(CC(=O)NC2CC3(CCN(C(C4CCCC5CC45)=O)C3)C2)cc2ccccc2n1 c1(OC)cc(-c2ccc(F)cc2C(=O)O)c2c(c1)CCO2 CN1C(Sc2ccccc2)CC1C(=O)NC1(C)CC(NC(C2(CF)CC2)=O)C1 c1(C(=O)NCCn2c(C)nnc2)cncc2nc(O)[nH]c12 N1(C(C(C)OCC(C)C)=O)CCCCC(NC(c2[nH]nnc2C2CC2)=O)C1 C1(CNC(C(C=C)(C)O)=O)CN(C)CCN1C(=O)Cc1ccnn1C1CCCC1 C12(CNC(=O)C#CC3CC3)CCC1CCN2C(=O)Cc1nc(-c2ccccc2)no1 N1(Cc2ncn(C)c2)CC2C(C(N3CCCC(C(O)C(F)(F)F)C3)=O)C2C1 Cc1cc(F)ncc1CCNC1(c2nnnn2C2CC2)CCC(O)CC1 N1(C(C(C)C#N)=O)CCC(CN(C(c2cccc(O)n2)=O)C2CC2)CC1 C(CNC(=O)C(c1cccs1)NC(=O)Cn1cc(CO)nn1)(C(C)(C)C)OC c1(C(N(CCCN(C(C2C(C=C)C2)=O)C)C)=O)sc2nccn2c1C c1(C(=O)NCC=CCNC(c2cc(-c3ccns3)on2)=O)ccncc1Cl C=CCCCCCC(=O)NC1CN(C(=O)CCCSC)CC1Cc1ccccc1 C1(CNC(=O)NC(c2cncc(C(F)(F)F)c2)CC(=O)OC)CCCC(C)(C)O1 C1(CC(C)C)C(=O)NCCC(OC)CNc2cc(ncn2)C(=O)N1.C(N)(=O)NC Cc1cc(C(=O)NC2CCCC2NC(=O)C(C)(C)c2ccns2)c(C)o1 C1(CC)C(=O)N(C)CCN1C(C1(NC(=O)C(C2CCC2)OC)CC(CO)C1)=O c1(C(=O)NCCNC(C(C)C)=O)csc(=NCc2c(O)cccc2O)[nH]1 C(=O)(C1CSc2ccccc21)NCC1CC(OC)CN1C(C1(C(N)=O)CC1)=O C12(CNC(c3nocc3Cl)=O)CC(C1)C(NC(C1CCSC1)=O)CO2 CCC(COC)(CC)C(=O)NCC(O)CNC(=O)CC(C)=C(C)C S(=O)(=O)(c1c(F)c(F)c(F)c(F)c1F)N1C(CN(C)C)CCCC1 N1(C(c2cnc(C(C)C)s2)=O)CC2OCCN(C(C3CCOC3C(C)C)=O)C2C1 Cc1occc(=O)c1OCC(=O)NCCC1CCN(C(c2cnn[nH]2)=O)C(C)C1 C1(C(=O)NC(CCOC)CNC(=O)Cc2[nH]cnc2C)CCn2c(O)nnc2C1 C1(CC(=O)NCCCCC2CN(C(=O)C=Cc3nccs3)C2)CCCC(O)C1 Cc1cn2cc(C(N3CCC(CCCCNC(C4CC4Cl)=O)CC3)=O)ccc2n1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2(C1)CN(C(=O)Nc1ccc(O)cc1)C2 c1(CN(C=O)CC2CCN(C)CC2)nnc2n1CCOC2 C1(C(=O)NC(CCSC)CO)CCN(C(=O)C2CC23CCCCC3)O1 c1(C(=O)NC(CNC(c2cc(C(CC)C)no2)=O)CO)ccc2[nH]nc(O)c2c1 N1(C(c2cnc(OCC)nc2)=O)CC2CC(NC(=O)COCCSC)C1C2 N1(C(C(CC(C)C)C)=O)CC(C)CN(C(=O)CCc2ccn(C)n2)CC1C N1(C(c2nc(C(C)C)sc2)=O)CCC(F)(F)C(CNC(c2snc(Cl)c2Cl)=O)C1 N1(C(C2CCC(C)C2)=O)CCN(C(=O)CCCS(C)(=O)=O)C2(CCC2)C1 Cc1cc(C)n(-c2ccc(NC(c3sccc3NC(C3(F)CCC3)=O)=O)cc2)n1 c1(C(N2CCCC(C(C(N3C(C)CCCC3)=O)(C)C)C2)=O)ncn2c1CCC2 Cc1cc(Cl)c(C(=O)NC2C=CCN(C(=O)CC(O)C(C)C)C2)nc1 CC(C(C)C(=O)NC1CC2(NC(c3ccnn3CCF)=O)COC1C2)S(C)(=O)=O C1(F)(CNC(CCCc2cc(C)no2)=O)CCCN(C(c2ncccc2N)=O)C1 c1(OC)cc(C(=O)NC2CC(N(C(=O)CN3CCC(O)CC3)C)C2)cc(N)c1 Cn1nccc1CC(=O)NC(CO)C(=O)NCC1C2CCCC12 CC(C)(O)C(=O)NNC(=O)c1cccc(S(=O)(=O)N2CCC(C)(F)C2)c1 N1(C(c2ccc(OC)s2)=O)CCN(C(=O)CNC(=O)CNC(C)=O)C(C(F)F)C1 N1(C(c2c(C)nc(CO)s2)=O)CCC12CN(C(=O)CSC(C)C)C2 C1(C(N(CC(N2CCOCC2)C)C)=O)COCCN(C(c2ccc(N)cn2)=O)C1 c1(C(=O)NCC2CC(O)CN2C(c2cn(C3CC3)nn2)=O)cncc2nc[nH]c12 c1(C(N(CC(CC)NC(C2CC(O)CN2C(C)=O)=O)C)=O)cnc2cccnn12 N1(C(Cc2cc(C)cc(C)c2)=O)CC2(CCC(CNC(=O)COc3ccsn3)O2)C1 CC1CCCN(C(c2coc(-c3ccccc3)n2)=O)C1CNC(C1COC1)=O CC(C)CCCCCC(=O)NC1(C2CCN(C(=O)C3=CCCC3C)C2)CC1 Cc1cn(C(C)(C)C(=O)N2CCC(NC(C3CCOC3)=O)C2)cn1 n1(CC)cc(C(C(=O)NCCN2CC(C)(C)C2)N(C2CCCCC2)C)cn1 C1(NC(c2c(C)onc2)=O)CC(NC(=O)C(N2CCSCC2)C)C(O)C1 C1(NC(c2nc(CCCC)sc2)=O)CCN(C(c2coc(C)c2)=O)C12CCC2 C1(CCNC(C2CCCC2O)=O)CCN(C(C2CCCCS2)=O)CC1(F)F C1(C(=O)NCCc2c(C)n[nH]c2)(NC(C2CC2C(N)=O)=O)CCN(C)C1 c1(CC(N2CC(c3cn(-c4ccccc4Cl)nn3)C2)=O)ccc(F)cc1 c1(C(=O)NC2CCN(C(C3CCCN(C(=O)OC)C3)=O)C2)nccc(C#N)c1F c1(COC)nc(NCc2cc(C)cc(Br)c2)cc(=NCCN2CCC(C)C2)[nH]1 c1(C(=O)NCC2C(NC(=O)CCCc3nccs3)C2)cc2ccc(F)cc2cn1 N1(C(C(C(C)C)(F)CNC(C2CCC(=O)N(C)C2)=O)=O)CCC12CCCOCC2 N1(C(c2ccc(C)s2)=O)CCC2(CC1)COC(CNC(C1CC(C#N)C1)=O)C2 C1(C(N2CC(NC=O)(CC)C2)=O)CCOCC1NC(=O)CCn1ccc(C)n1 c1(CNC(C(c2cc(C)oc2C)NC(=O)OC(C)(C)C)=O)ccc(C)c(C)c1Cl CC(C)C(C(=O)NC1CC(F)(CNC(=O)CC2CC2(Cl)Cl)C1)NC(N)=O CC(C)CC(O)C(=O)N1CCCC1C(=O)NCc1sccc1CO C1(CC(=O)NCC(CC)NC(c2snnc2CC)=O)CCCC(OC)C1 C(=O)(C(CCNC(C1CCCCS1)=O)N(C)C1CC1)N1CC(O)(CCN(C)C)C1 c1(NC(=O)NCC2COCC2N2CCCC2)ncc(C(F)(F)F)s1 N1(C(c2cc(C)oc2C)=O)CC(C)C(NC(=O)CCc2ccsc2Cl)C(C)C1 Cc1nnn(C)c1C(=O)NCC1CCCC(NC(=O)C(C)(C)c2ccccc2)C1 C1(N(C(=O)CCCc2cncs2)CC)CCCN(C(=O)C(COC)CC)C1 N1(C(C2(CNC(c3cc(C4CC4)on3)=O)CCOC2)=O)CCCOCC1 Cc1ccc(F)c(C(=O)NCC2(F)CCC(NC(c3cc(C(F)F)[nH]n3)=O)C2)c1 c1(C(=O)OC)coc(C=CC(N2CC(NC(=O)CC3CCC4CC4C3)CC2C)=O)c1 Cc1c(C(=O)NC2(CO)CCN(C(=O)COc3cccnc3)C2)cccc1O N1(C(c2sc(CC)c(C)c2)=O)CCC2(C1)CN(C(C1(C(N)=O)CC1)=O)CC(C)O2 c1(C(N(C)CCOCCNC(C2CCCC2F)=O)=O)cc(=O)cc[nH]1 Cc1cc(C(=O)NC2CC(NC(c3cnco3)=O)C2)c(F)c(Br)c1 C(C(C(=O)N1CCN(CC(C)O)CC1)C(C)(C)C)N(C)CC.C1=CCNC1=O N1(C(C)C(=O)NC(CO)C(C)NC(=O)C=Cc2nccs2)CCCCCC1 N1(C(c2c(COC)noc2)=O)CCC2(NC(c3nn(C)c(C)c3Cl)=O)CC2C1 C1(C)(CC(=O)NCC=CC(=O)NC(C)C(C)OC)OCCO1 c1(CC)nccc(N(CC(C)CNC(=O)CCc2cc(C)no2)C)n1 C1(C(=O)NC2(CNC(CC(C)(C)O)=O)CCOC2)COC2(CCC2)CO1 c1(C(N(C)CCOCCNC(=O)C(F)C2CCCO2)=O)cnoc1-c1ccco1 C1(C(N2CCC(C=C)C2)=O)COC2(C1)CN(C(=O)C#CC1CC1)C2 N1(C(CC=C)=O)CCN(C(c2c(C)cc(C#N)cc2C)=O)CC12CCC2 c1(NC(C(CC)(C)O)=O)ncc(C2=CCC(C)CC2)cc1C c1(C(=O)OC)cc(C)c(NC(=O)C(=O)NCC2CC(CO)CO2)cc1F.C1CC1 C1(C(=O)NC2(CC)CCCC2)CN(C(=O)C(=O)NOC)C2(CCC2)C1 CCCCC(O)C(C)C(=O)N1CC(C(=O)NC2CN(CC(F)F)C2)CCC1C C1(NC(Cc2c(C)n(C)nc2)=O)COCCN(C(c2nc(O)[nH]c(=O)n2)=O)C1 N1(C(C(=O)NC2C(C(=O)OCC)CCCC2)=O)CCC2(CCCNC2)C1 CCCCC(=O)N(C)CCN(C)C1CC1.C1(S)CCCO1 N12CC3CCN(C3C1)C(=O)C1(c3ccc(cc3)C2=O)CC1.c1(OCC)cocn1 c1(CC(=O)NCC(C)N(C)C(C2CC(C#N)C2)=O)cc(Cl)ccc1Cl c1(C(=O)NCCCNC(C(CSC)OC)=O)cn(C)nc1C c1(CNC(C(N2CCCC3CC23)C2CC(CC)C2)=O)cc(F)ccc1F N1(C(C2CCN(CC)C2)=O)CC(NC(C2(CCOC)CC2)=O)C(C(F)F)C1 c1(C(=O)NCCCSCC(=O)NC2CCN(C(=O)COCCF)C2)cccnc1 c1(CNC(COCC)=O)cn(C)nn1.C1(C)CN1C N1(C(C(C)OC2CCOCC2)=O)CCCC12CCN(C(c1ccc(O)nc1)=O)CC2 c1(-c2cn(CC3CCN(C(c4ncn(C)c4)=O)C3)nn2)cnc2cccnn12 c1(C(C(=O)NCCC2CC2)N(C2CCCC2O)CCC#N)cccc(Cl)c1Cl C12(C(N3CC(c4ccon4)C3)=O)CCCC1CN(C(C13CCC(CC1)C3)=O)C2 C1(F)(C(N(CCCCN(C(=O)C(F)n2ccnc2)C)C)=O)CC=CCC1 N1(C(C2COCCC2(O)CO)=O)CCOCc2cccc(Br)c21 C1(C(=O)NCCCN(C(c2cccc(CF)c2)=O)CC)CCCC(N(C)C)C1 C12CCC(CC1)C(=O)N2.c1(-c2cn(C3(C(=O)OC)CC3)nn2)nccc(C)n1 C(=O)(CC(CNC(=O)N(C)C)C1CC1)NCC1CN(C(C)C)C1 c1(C(=O)NC2CC3N(C(C(CC)(C)C#N)=O)C(CC3)C2)cnc2ccnn2c1C c1(C(N(CC(CN(C(c2c(COC)nn[nH]2)=O)C)O)C)=O)cnccc1N(C)C C(=O)(C(C)(C1CC1)N(C(=O)C(c1ccnn1C)O)C)NC(C1C(C(=O)OC)C1)C C1(CNC(c2nc(CS(C)(=O)=O)sc2)=O)CC2(CCC2)CN1C(=O)C1=CCCC1 c1(C(=O)NC(CC=C)CNC(=O)CNS(=O)(=O)C2CC2)[nH]nc([N+](=O)[O-])c1Cl c1(CC(C(=O)O)NC(CCNS(CC)(=O)=O)=O)ccc(OCC)c(F)c1 c1(C(N(C)CCSC2CC(=C3CC3)C2)=O)cc(S(N)(=O)=O)co1.C12(CC1)C(=O)NC2 C(=O)(C(C(C)NC(c1ccnn1CCF)=O)C(C)C)Nc1cccc(COC)c1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(CC)C(N1CC2(CCCC2)C1)=O C(=O)(CC(=O)OC(C)(C)C)NC(CNC(C(C)NC(CC)(C)C)=O)Cn1cccn1 CN1CCC(NC(=O)C(C2CCCC2)NC(=O)COC2CCCCC2)C(C)(C)C1 C12(NC(c3c(C)n(C)nc3)=O)CCCC1N(C(c1cc(O)ccc1O)=O)CCC2 CC(CCCCO)NC(C1CC1C(C)NC(=O)CC1COCCOC1)=O CN1CC2(CCN(C(c3cc(NCc4ccc(Br)c(Cl)c4F)cn3C)=O)CC2)C1 c1(C(N(C)CC2CN(C(c3ccn(CC)n3)=O)C2)=O)c2n(c(=O)n1C)CCCC2 C1(C(N2C(C(=O)NCC(c3ccncc3)C)C=CC2)=O)CC12CCCCC2 N1(C(C2C(C)C2)=O)CC2(CCC(CNC(C3C(C)(C)C3(F)F)=O)O2)C1 N1(c2cc(C)[nH]n2)CCN(C(c2cncn2C(C)C)=O)CC1 C12(NC(C=Cc3scc(C)n3)=O)CCCC1CN(C(C1CCOCC1)=O)C2 c1(OC)ccncc1CC(=O)NCCCC(C)NC(c1cnsc1)=O C1(C(N(CC(=O)NCC2(OC(C)C)CC2)C2CCC2)=O)CC2OC1C1CC21 C1(N(C(C(F)=CC)=O)C)CCCN(C(C2CC(=O)N(C)C2)=O)CC1 c1(CC)nn(C)cc1CNC(=O)C(Cn1cccn1)NC(=O)Cc1cc[nH]n1 C(=O)(C(C#N)CC1CC1)NCC(CCC)NC(c1oc(C2CC2)nc1C)=O CCS(=O)(=O)CC(=O)NCC1CC2(CC2)CN1C(c1scnc1C1CC1)=O c1(CC)nccnc1C(=O)NCC1(F)CN(C(C2CN(C)CCO2)=O)C1 Cc1coc(C)c1C=CC(=O)NC1CCC(CNC(c2cnn(C(C)C)n2)=O)C1 c1(C2(NC(=O)CC3CCN3C(=O)CN3CC(=O)NC3=O)CC2)cc(CO)ccn1 C=CCCCCC(=O)N1CCCC2(NC(=O)CCNS(C)(=O)=O)CC2C1 N1(C(C(C=C)C)=O)CC(C(N2CCC(CO)(CO)C2)=O)C(F)(F)C1 C=CC(C)(CC)C(=O)NC(C1CN(C(=O)CCn2cc(Cl)cn2)C1)C CCCCCC(C)CC(=O)N1CC2CC(C1)N(C(c1[nH]nc(OC)c1Cl)=O)C2 N1(C(CNC(CCC)=O)=O)CCN(C(c2cnn(C3CCC3)c2)=O)CC1C1CC1 C(CCSC)(C(=O)NCC(C1CCC1)CC)NC(c1ccccc1COC)=O C(=O)(C#Cc1ccccc1)NC(c1ccc(OC)cc1)c1noc(C)n1 Cc1[nH]nc(C(=O)NC(C2(CNC(c3cnn(C)c3C3CC3)=O)CC2)C)c1Cl CC1CN(C(=O)C(CO)NC(N)=O)CCN1C(=O)CCCC(=O)N(C)C C(=O)(CCC(=O)NCc1ccc(NC(C2CCN(C)OC2)=O)nc1)NCCC c1(C(=O)OC)oc(C(=O)NC(C)CNC(=O)CSc2ccc(F)cc2)cc1C c1(C(=O)NCCC)cnc(O)c(NC(=O)Nc2ccc(N(C)C)cn2)c1 C(CS(=O)(=O)NCCCC(C)NC(=O)C(=O)NCCNC1CCCC1)OCC.OC c1(COC(C)C)ccc(NC(C)C(=O)NC2CCCCO2)nc1 Cc1ccc(C(=O)NC2COCC2NC(c2cc(F)n(C)n2)=O)c(Br)c1F C1(C(N2CC3C(NC(=O)COCC4CCOC4)C3C2)=O)CC2CCCC2C1 C(C(C(=O)N(CCF)C1CC1)NC(c1cc(OC)ns1)=O)OCC c1(C(N(C2CCCN(C(c3cc(Cl)cnc3O)=O)C2)C)=O)ccc(Br)c(Cl)c1F C(=O)(C1=NNC(=O)CC1)NCC(C)NC(CC(c1c[nH]c2ccccc12)C)=O C1(C2(N(C)C)CCC2)(NC(N(c2ccc(Cl)cc2)CC)=O)CCC1 C(C(=O)N1CCC1CNC(=O)C(C)(C)n1cnnn1)(C(C)(C)C)OC c1(C(N2C3CC(NC(C(C)O)=O)C2CC3)=O)c[nH]c2nccc(Cl)c12 c1(CNC2=NCc3ccc(cc3)CN2)cn2ccsc2n1.C1(CSC)CCCO1 c1(C(=O)NCC(F)CNC(=O)C(F)CC2CCC2)cc(-c2ccncc2)on1 c1(C(N(C2CC(NC(C(COCC)C)=O)C2)C)=O)ccc(F)c(CC)c1 C1(C(=O)NC(C)CN(C)C(C2CC(F)(CF)C2)=O)CCc2nc[nH]c2C1 c1(C(N(CC(=O)NCC23CCC(CC2)C3)CCOC)=O)ccc(C#N)cc1 c1(C(=O)NCC2(F)CCC(NC(C3CCN(C(C)=O)C3)=O)C2)cc2cnccc2o1 N1(C(CC=C=C)=O)CC2CC1CN2C(=O)CN1CCC(F)(F)C1 C#Cc1cccc(CNC(=O)C(CC2CCCC2)NC(c2cnnn2C=C)=O)c1 C#Cc1ccc(C(N2CCC(C(=O)Nc3cc(OC)ccn3)C(O)C2)=O)c(Cl)c1 N1(C(c2c(OC)noc2C)=O)CCC(CNC(=O)C(F)F)C12CCC2 c1(C(=O)NC(C2CN(C(=O)C3=CC(C)(C)C3)C2)C)ccc(Cl)c2cccnc12 c1(C(N2C(CNC(C(CO)N(C)C)=O)C=CC2)=O)cc(Cl)c(Cl)cc1N CC(Cc1ccc(Cl)cc1)CC(=O)NC1CC(NC(c2nocc2C2CC2)=O)C1 N1(C(C2CN(C(c3cnn(CC)c3C)=O)CC2(F)F)=O)CC2(CCC2)C12CCC2 C1(CCNC(=O)C=CCO)CCCN(C(=O)CCC(=O)c2cccs2)CC1 N1(C(C(CC#C)C)=O)CCC2CCN(C(c3nccc4[nH]ccc34)=O)CC12 CCC(C)(C)C(O)C(=O)N1CC2(C(N3CC4CCC3C(OC)C4)=O)CC1CO2 CC(C)C(CNC(=O)C(C1CC1)C1CC1)C(=O)NCC(C)(C)C1CCCC1 CCC(O)C(F)(F)C(=O)NCC1(F)CC(Nc2ncnc3[nH]cnc23)C1 O=C(C1=NOC2COCC12)NC1(C2CCCCN2C(=O)CN2CSCC2=O)CC1 c1(C(C(=O)NCCC)N(C)Cc2nc[nH]n2)cc(OC)c(OC)c(F)c1 CC1CN(CC2CC2(Cl)Cl)CCc2cc(Br)c(O)cc21 c1(OC)cc(F)c(F)cc1C(=O)NC(C)C(C)NC(c1cocn1)=O CC1CCN(C(=O)CCC2NC(=O)NC2=O)CC1NC(c1cncc(Cl)c1Cl)=O N1(C(c2cc(CCNC(c3c(C)ccc(F)c3)=O)on2)=O)CCC2(C1)CC2(F)F N1(C(CCOCC)=O)CC23CCCCC2(C1)CN(C(c1ccc(Cl)cc1F)=O)C3 Cc1cc2n(n1)CCN(c1ncccc1S(=O)(=O)NC1CCCC(F)(F)C1)C2 c1(C(N2C(C(C)(C)NC(CCOCCOC)=O)CCC2)=O)ccc(F)c(Cl)c1F CN1CCCC1=NS(=O)(=O)c1cccc(NC(=O)CC2CC2C(F)(F)F)c1 c1(C(=O)NC(Cc2ccccc2Br)C(=O)NC2CC2)ncccc1Cl CS(=O)(=O)c1ccc(C(N2CCC(NC(c3ccccc3CO)=O)C(O)C2)=O)[nH]1 Cc1nc2c(cc1C(N1CCC(CNC(C3(F)CC3)=O)C1(C)C)=O)CCCN2 CC(C)CC(C)CC(=O)NCC1CN(C)CCN1C(c1cc2c(s1)CCSC2)=O c1(CCC(=O)Nc2ncc(C)s2)ccc2c(c1)OCCO2.C(CC)N(C(=O)C)C C12(C(=O)OC)CCCC(C(N3CC4C(NC(=O)C(Cl)=CCl)C4C3)=O)(CC1)C2 Cc1ccc(F)cc1C(=O)C(N1CCCC1CNC(=O)CSC1CCCCO1)=O N1(C(C(CC)SC)=O)CCC(C(C)NC(c2cnn(CC)c2C)=O)CC1 c1(C(C(N2CC(N(C(CC=CC=C)=O)C)C2)=O)OC)ccc(F)cc1 N1(C(CC(C)Nc2cncn2-c2ccccc2)=O)CCN(CC(C)C)CC1C C1(CNC(Cc2cccc(C)c2)=O)CN(C(=O)CC(C)P(C)(C)=O)CC12CCC2 C.C(=O)(CC(=O)N(CC)CCCCOCCOC)N(CC(N(C)S(N)(=O)=O)=O)C.OC c1(NCC2C3CN(C(c4n(C)nc(CC)c4Cl)=O)CC32)ccc2n[nH]cc2c1C C1(CN(C)C(C2N(C(=O)CCC3CCC3)CCC2(C)C)=O)CCCCC1(C)C C1(C)(CNC(C=CC(C)(C)NC(CCc2n(C)ccc2)=O)=O)CC2CC2C1 C1(OC)CC(NC(=O)CCCC#N)CN(C(c2ccn(C)n2)=O)C1 C1(NC(C2(OCC)CCC2)=O)CCCC1CNC(C1CCN(CC(F)(F)F)C1)=O C12(C(=O)NCC(C(C)C)NC(Cc3c(C)cccc3C)=O)CCC(CC1)C2(C)C N1(C(C)=O)CCN(C(=O)Nc2sc(OC(C)C)nc2C)CCC1C CC1(C)CCC(C(N2CC(n3c(O)nnc3O)C2)=O)CN1C(=O)CC(F)(F)F C1(NC(CSCC#C)=O)CCN(C(c2cc(CC)ccn2)=O)CC1C(C)C C(N=c1nc(N2CCCC(C)(N3CCC3)C2)c2ncn(C)c2[nH]1)C1(CC(C)C)CC1 Cc1nc(NCC2CCCCC2NC(=O)Cc2cc(C3CC3)no2)cc(O)n1 N1(C(c2cc(C)c(F)cc2N)=O)CCCC2C1CCCN2C(=O)Cc1cccs1 C=CC(C(=O)N1CC=CC1CNC(c1ccncn1)=O)c1ccccc1 N1(C(Cc2c(C)cccc2)=O)CC(C(N2CC3CC2CN3C)=O)C(C2CC2)C1 N1(C(C2(OC)CC2)=O)CCC2(CCC(NC(=O)CC3CC(F)(F)C3)C2)CC1 C1(CN(CCOC)C)CCCCN1C(c1cccnc1)=O.C(C)(=O)O c1(C(N(C2C(OC)CCCC2)CC2CCOCC2)=O)c(N)c(C(F)(F)F)nn1C CC1=CCC(C)(C(=O)NC2CC3CC2N(C(c2cccc(C(F)F)c2)=O)C3)CC1 C12CCN(CC1C)C(=O)COCC(=O)N2.C(C(=O)NCCOC)N(C)CC C1(CN(C(Cn2c(C)ccn2)=O)C)CCCN(C(=O)C=CC2CCCCC2)C1 C1(NC(c2c(C)[nH]cc2)=O)CCCCN(Cc2cn(-c3ccccc3Cl)nn2)C1 C(=O)(C(C)(C)CN(C(=O)CC(C)CN(C)C)C)NCc1ccc(SC)o1 N1(C(CN(C2CC2)CC)=O)CCC2C(C1)CN2C(=O)C(c1cccn1C)=O N(C(=NCCCCC(F)(F)F)NCC(C(F)(F)F)n1cccn1)CC(C)C(C)(C)C C1(C)(C(=O)NC2(CC=C)CCN(C(=O)CN3CCCNC3=O)C2)CCC(C)CC1 C1(C(N2CC3C(CNC(=O)CNC(C4CCC4)=O)(C3)C2)=O)CCc2nncn2C1 C(C)(CCC(=O)N1CC(C)C1C(=O)NCC1CCCS1)OC N1(C(C(C)S(N)(=O)=O)=O)CC(C)CC(C)(C)C1.c12nc(co1)C(=O)NOC2 C1(OC(CC)=O)CCN(C(=O)CCC2(C)CN(C(c3cc(OC)cs3)=O)C2)C1 Cc1ccc(NC(=O)C(F)C2CC(NC(=O)CCc3ncccn3)C2)cc1F C1(CCc2ccccc2NC(C)=O)(NC(=O)NCC)CCOCC1 C1(C(=O)NC2CCN(C(C34CC5CC3C4C5O)=O)CC2)CCC2(CCC2)CO1 c1(CCCC)ccc2nc(C(=O)N(C(c3ccccc3Br)C(=O)O)C)oc2c1 N1(CCC)CCCCC1C(=O)NC1CN(C(c2cc(C(C)(C)C)c[nH]2)=O)CC1F c1(C(N(CC(CN(C(C(CC)NC(C)=O)=O)C)O)C)=O)ccn(C2CC2)c1C c1(C2C(C)=NN(C)C2=O)nc2c(s1)CN(CCc1ccccc1)CC2 C=CCC(CNC(C1CCNC1=O)=O)C(=O)Nc1cn(C)nc1OC N1(C(CC)=O)CCCC(C2CC2NC(=O)C2COc3ccccc32)C1 c1(C(=O)NCC(CNC(C(C)NS(CC)(=O)=O)=O)(C)O)cc(O)nc(O)c1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2CN(C(C3CCC(=O)N3)=O)CC2C1 C=C(C)CCCC(=O)NC1C2CC1N(C(c1ccc(Br)o1)=O)C2C c1(C(N2C(C)CC(NC(c3nc(CC)oc3)=O)C2)=O)cc2ccccc2c(=O)o1 C1(C2CN(C(=O)CCc3cccnc3)C2)(NC(=O)CCn2cnnn2)CC1 CCCC(O)C(=O)NCC(CNC(=O)Cc1cn(C2CC2)cn1)CO C1(NC(CC(C)C)=O)CCC2(CC1)CC(NC(c1cc3c([nH]1)CCCC3)=O)C2 N1(S(CC)(=O)=O)C(C)CN(c2nc(C)ccc2OC)CC1C C(C)(C(=O)NCCOC1CCN(C(c2c[nH]nc2C)=O)C1)(C1CC1)OCC c1(C(=O)NCC(C)CN(C)C(c2cn(C)nn2)=O)nn[nH]c1Cl C1(N(CCCC(N)=O)C(=O)Cc2ccccc2O)CCCC12CCNCC2 C12(C(=O)NC3C(C(=O)NC4(CC)CCCCC4)COC3)CCC(C1)OC2C N1(C(CNS(CC)(=O)=O)=O)CC(CNC(=O)CCC(CC)OCC)C2(CCC2)C1 c1(C(c2nc(CC)no2)N(C(=O)NCCOC(C)(C)C)C2CC2)ccccc1Cl C1(N(C(c2ncc(CC)cn2)=O)C)CCCCN(C(=O)CNc2ccccc2)C1 C(N=C(NCC(F)(F)C(F)(F)F)N1CCC(O)CC(C)(C)C1)c1nc(CC)[nH]n1 c1(C(=O)NCC(C2CC2)NC(c2c(CCC)cccc2)=O)cc2c(s1)CC(O)C2 CC1CCN(C(=O)C#CC(C)(C)O)CC1NC(=O)CCCNC(N)=O C(=O)(C(F)CC(C)C)NC(C1(O)CN(C(CCCc2onc(CC)n2)=O)C1)C CN(C)NC(=O)CCC(=O)NC1CCC(CCC(=O)NC2(C(N)=O)CCCC2)C1 C#CCC(CC#C)NC(=O)CCC(C)NC(=O)C(C)C C(=O)(CS(=O)(=O)CCO)NCC1(C(N)=O)CN(C(C2CCOC2C2CC2)=O)C1 CCCCC(O)CC(=O)NC(C(=O)NCC(C)(O)CCO)C(C)CC CCC(CCC(=O)N(CCOC)C(C)C1CC1)NC(=O)C(F)n1ccnc1 C(C(C)C(=O)NC(C(C)(C)CCCCN(CCC(=O)N)C)C)OCC.N(C)C N1(CC(=O)NC2CC(C(=O)NCC(C)(C)F)C2(C)C)C(=O)CCCC1=O Cc1cnc2n1CCN(C(C1CN(C)CCN1C(=O)COCCF)=O)C2 N1(C(C(C)(C)OC)=O)CC(CNC(c2cnc(C3CC3)o2)=O)C(F)(CO)C1 C(=O)(C1=CCCCC1C)N1C(C)CCC(NC(c2c(CC)nc[nH]2)=O)C1 C1(S(C)(=O)=O)(C(=O)NC2C3(CN(C(C#CC(=O)N(C)C)=O)C3)CC2)CCOCC1 c1(C(=O)NC2CC(C)CN(c3ncc(C#N)cc3Cl)C2)cc2ccccn2n1 C(C(C)C(=O)N(CC(C)N(C(=O)CSc1nccn1C)C)C)OCC C1(C(=O)NCC(C)(CO)NC(c2c(C)csc2)=O)CCN(C)S1(=O)=O N1(C(C2(C)CC2)=O)CCCOC(CNC(=O)CC2CSCCS2)C1 C#CCC(C)(C)C(=O)NC1CC=C(C(=O)N2CC(C)(C)C2COC)C1 C1(NC(CN(S(C)(=O)=O)C2CC2)=O)CN(C(=O)CC2(C3CC3)CC2)C(C)(C)C1 C(=O)(C1=NN2CCCN=C2N1)NCC=NC(=O)CSCc1cccs1.C12CC(C1)C2 C1(=CC(=O)NCC2C(NC(C(C)=C3CC3)=O)C2)CCC(C)CC1 C#Cc1ccc(C(=O)NCCC(C)(C)NC(c2cccc(C3CNC3)c2)=O)o1 C1(CC)CN(C(C2CC(CCNC(=O)CC3=CCCC3)C2)=O)CCN1C N1(C(COCC(=C)C)=O)CCC(CO)(CNC(c2ccc(F)cc2F)=O)CC1 c1(OC(c2snc(OCC)c2Br)=O)nc(NC(=O)OC)c2n1CC(C)CC2 CCCCC(O)CCC(=O)NC1CN(C(c2sccc2C(C)C)=O)CC(C)(C)C1 c1(C(=O)Nc2ncccc2Cl)cn2c(n1)CN(C(=O)Cn1ccnn1)CC2 C(C(=O)NC(CN(C)Cc1nccs1)Cc1ccccc1)(C(C)C)OCC(C)C c1(SCC(=O)NCCCCNC(C2CC3CCC2O3)=O)ccc(F)cc1F C(=O)(CC(F)(F)C(F)F)N1CC(NC(C2(c3cc[nH]n3)CC2)=O)CC(OC)C1 N1(C(C(C)N2CCC2)=O)CC(CNC(=O)CSCC(F)(F)F)CC12CCOCC2 n1(CCC)ncc(C(=O)NCC2CC(NC(C3(CO)CCCO3)=O)C2)c1C1CC1 C1(C)(NC(C(C2CCOCC2)OCC)=O)CCN(C(=O)C=Cc2cncs2)C1 c1(OC)cc(C(=O)NCC2CC2NC(c2cocc2CN(C)C)=O)ccc1OC C(=O)(CC1=CCN(C)CC1)N1CCC(CNC(C(C)(C2(C)CC2)OC)=O)CC1C Cc1[nH]c(C#N)cc1COc1ccc(CNC2CCCC(C)CC2)cc1 C(=O)(C#CC1CCCCO1)N1CCC(NC(C2C3CCCC23)=O)C(F)C1 CCC(CN=c1ccc(S(=O)(=O)N2CCCOC(COC)C2)c[nH]1)OC c1(CNC(C2CN(Cc3cncnc3)C2)C)cnc(O)c(C(=O)O)c1 CC(CN(C)C)CCC(=O)NC(C)(CNC(c1nn(C)c(Cl)c1Cl)=O)CO c1(C(N2CC(C)C(NC(c3ccn4ccsc34)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 C#CCCC(O)C(=O)N1CCOC(C(C)NC(c2cc(N)ccc2Br)=O)C1 C1(CN(C(c2ccc(C(N)=O)o2)=O)CC)CCCCN1C(C1COC(=O)C1)=O C(=O)(CCCC(F)(F)CO)NCC(C(C)C)NC(Cc1n[nH]c(=NCC)s1)=O N1(C(C=C(C)C)=O)CCC(O)(C2(C(=O)NCCF)CCOCC2)CC1 c1(CC(N2CC(NC(C(CC(C)C)=O)=O)C(C)C2)=O)noc2ccccc12 N1(C(Cc2c(OC)cccc2)=O)CC(C)CN(C(C2CC2(Cl)Cl)=O)CC1C n1(CC)cccc1C(=O)NC1CCCC1CNC(C1CCS1(=O)=O)=O c1(CN(C)C)ccc(C(N2CCC(N(C(=O)CNc3ccccn3)C)C2)=O)cn1 c1(C(=O)NC2C=CC(CNC(=O)CCn3cccn3)C2)cc(C2CCOC2)[nH]n1 N1(C(c2c(CC)nco2)=O)CCN(c2nnc(C)s2)CC1 n1(CC(=O)NCC(c2ccc(CC)cc2)OC)cccc(C)c1=O C(=O)(CCCCCNC(C1(OC)CCC1)=O)NCc1c(CC)nn[nH]1 C1(NC(Cc2ncn(C)n2)=O)CC(CC(=O)NCC2(C3CCC3)CC2)C1(C)C C(=O)(CC1=CCCC1)NCCCCC1(NC(c2cc(C)no2)=O)CC1 N1(C(C(CCNC(=O)C(F)C(F)(F)F)OC)=O)CCOC(C)(C)C1C CCCCC(CNC(=O)CCc1cccc(C(F)(F)F)c1)NC(c1nncs1)=O c1(C(N2CCC3CC23C(=O)NCCF)=O)cc(F)cc(F)c1 c1(OC)cc(NC(c2ccnc(CNC(=O)C(C)(C)F)c2)=O)cc(C#N)n1 N1(C(C(CCC)NC(N)=O)=O)CC2CC(NC(c3cc(C)nc(O)n3)=O)C1C2 C1(C(C)NC(CN(C(C)=O)C)=O)CCCN(C(=O)C=CSC2CCCC2)C1 N1(C(c2c(C)n(C(C)C)nc2)=O)CCC2(CCCN2C(C2CCCSC2)=O)C1 N1(C(c2c(OC)c(C)ccc2)=O)CC(C)OC2(CCN(C(=O)CCCC#N)C2)C1 Cc1nn(C)c(Cl)c1CC(=O)NCC1C(C)CCN1C(=O)C=Cc1cccs1 CN1CCC(C(=O)N(CCCCNC(=O)CC2CC2)Cc2nnnn2C2CC2)C1 N1(CC)N=C(C(=O)NC2(COC)CCN(C(=O)C=C(C)C(C)(C)C)C2)CCC1=O c1(SC)cc(F)ccc1C(=O)NCCCCCN(C(=O)CSc1nnnn1C)C CC(CNC(C1(CO)CCCN(C(=O)C(O)C(F)(F)F)C1)=O)CC(F)(F)F Cc1cccc(CC(=O)NCC2CC(CNC(C3CC(O)C3)=O)CO2)c1Br C1(CNC(C=CCCC)=O)CN(C(c2ccc(C)c(Br)c2)=O)C(C)(C)C1 C1(NC(C(C=C)(C)C)=O)CCN(C(=O)Cc2ccsc2)C12CCCC2 S(=O)(=O)(c1cc2nc(O)[nH]c2cc1Br)N1C(CC2(C)CCCO2)CCC1 C(CCCCCCCSCC(F)F)(C(=O)NC1CC1)NC(CC(C)(C)C)(C)C#N C1(C#N)(C(=O)NC2CC(N(C)C(C3CC(n4ccnc4)C3)=O)C2)CC2CCC1CC2 c1(OC)cc(OC)c(S(=O)(=O)N(CCO)Cc2ccc(F)cc2)c(OC)c1 C(=O)(C(CCF)NC(c1nccnc1N)=O)NC(c1onc(C)n1)C C(=O)(CC1CCCc2ccccc21)NCC(C)NC(C1(C)CCC(=O)CC1)=O N1(C(C(CCC)NC(=O)C(C)OCOC)=O)CCN2CCCCC1C2 c1(C(N2CCC(CCC(=O)NC3(C(=O)OC)CC3)C2)=O)[nH]cc(C)c1C C1(C(N(CCCNC(=O)CC2CCCC2)C2CC2)=O)C2CCC1(c1ncco1)C2 N1(C(CCCCN(C)C)=O)CC2CCN(C(C3CCn4ncnc4C3)=O)CC2C1 C(=O)(C#CC1CCC1)NCC1(F)CCN(C(C(c2ccc(F)cc2)C)=O)C1 C(C(C)(C)C(=O)NCCC1CC1C)NC(C(C)=C(C)C)=O c1(OCC)ccc(C)nc1C(=O)NCC(C)(CC)NC(c1coc(C(N)=O)c1)=O Cc1c(C(N2CCCC(C(=O)NOCCC(F)(F)F)C2)=O)ncn1C N1(C(c2c(Cl)cnc(CC)n2)=O)CCCC2CN(C(C3C4COCC34)=O)CCC12 Cc1ccc(C(C)Oc2sc(C(N3CC4C(C(=O)NCC)C4C3)=O)c(C)n2)cc1 C1(C2CN(C(c3ccsn3)=O)C2)(NC(c2ccc(OC)cc2)=O)CC1 Cc1cncc(CC(=O)N(C(C)CN(C)C(C2CC23CCCC3)=O)C)c1 Cc1cccc(F)c1CC(N1CCCC(NC(=O)C=Cc2cc[nH]n2)C1C)=O N1(C(c2cc(OC)c(N)cc2)=O)CC(NC(C)=O)C2CCCCC12 CC(C)CC(C)CC(=O)N1CCCC1C(N1CC2(CCCC2)C1)=O C=Cc1ccc(CNC(C2CC2C(=O)NCCc2ccc(F)c(Br)c2)=O)cc1 N1(C(C=CC(C)NC(C(C(CC)CC)OC)=O)=O)CCCC12CCOC2=O C1(NC(CCN(C(c2cc(OCC)n[nH]2)=O)C(C)C)=O)CC2(CCC2)C1O C1(CC)CC(C(=O)NC2(C(C)NC(=O)C(=O)NC(C)C)CCC2)CCO1 c1(CN2CC3(C(C(=O)Nc4c(I)ccc(OC)c4)C3)C2)cc(F)c(F)cc1F C1(NC(=O)COc2cccc(F)c2F)CN(C(=O)CCF)C2(CCOC2)C1 c1(C(C)N(CCn2cccn2)CC2CC2C(F)(F)F)cccc(C2CC2)c1 N1(C(c2c(N)cn(C)n2)=O)CCC2(COC(=O)N2)C1 c1(C(c2n(CCC3(C)CC3)nnn2)NC2(C)CCSC2)cc(Br)c(F)cc1F C1(NC(N(CC#Cc2ccccc2)C)=O)CCN2CCCCC12 C#Cc1ccc(C(=O)N(C2CN(C(=O)C(C)CC(C)(C)C)CC2O)C)cc1F C1(COC)(NC(c2ccn(CCO)c2C)=O)CCCCC1.C1(=O)N(C)CCN1 N12CCCC1C1CCCCN1C(=O)c1nnsc1C2=O.c1(CC)csnc1OC CCCCCCCCC(=O)NCC1CCN1C(c1nsc2ccc(C)cc12)=O N1(C(C2CC23CCOC3)C(=O)NCCCCCCCC)CCCCC12CCN(C)C2 O=S(=O)(c1c(OC(F)(F)F)cccc1Br)NCc1cccnc1 N1(C(COCc2c(C)ncs2)=O)CCCC(C)(C)C1CNC(=O)C(C)(C)C c1(C(=O)O)ccccc1.C12CC1C(=O)NCCCCNC(=O)CCN2 c1(C(N2CC(NC(c3csc(C(F)(F)F)c3)=O)C(O)C2)=O)cnc2ccsc2c1 N1(C(C2C(OC)CCC2)=O)CCCC(NC(C2CCC(=O)N2)=O)CCC1 C1(CN(C(COC)=O)C)CCN(C(c2n[nH]cc2C2CC2)=O)C1 N1(C(c2c(C)sc(Br)n2)=O)CCC(C)C(CNC(c2coc(O)n2)=O)C1 Cn1nc(C(N2CCOC(C)(CNC(c3c[nH]nc3F)=O)C2)=O)ccc1=O CCS(=O)(=O)Cc1cn(CC2CCCN2C(C2(C)CC2C)=O)nn1 C12(C(=O)NC3C=CCN(C(C4CC(N5CCCC5)C4)=O)C3)CCN(CC1)CC2 N1(CC)C(=O)CC(C(=O)NCC(C)C(=O)NC)C1c1ccc(OC(F)F)cc1 N1(C(c2cnc(OC)nc2)=O)CCCC(C)C1CNC(c1ccc(C)c(O)c1)=O c1(NC(C2(C)CN(C(=O)CC#N)C2)=O)cc(CO)ccc1Cl CC(CCS(C)=O)NC(c1ccnn1C1CNC1)=O N1(C(CC(C(F)F)NC(c2nccc(OC)c2)=O)=O)CCOc2ccccc21 c1(C(N2CCC(SC)C2)C(=O)NCCC#N)ccc2c(c1)OCCO2 C1(NC(C2ON=C(CC)C2)=O)Cc2ccccc2C1 C(=O)(C1=Cc2ccccc2C1)NCC1(C(=O)NCc2nc(CC)n[nH]2)CC(=C)C1 c1(CN2CC3N(C(Cc4c(C)noc4C)=O)C3C2)cc(Br)cc(Br)c1 C(=O)(C(C)(C)C(C)O)NCC(C)CNC(=O)Cn1cccnc1=O N1(C(C(C)O)=O)CC2CCN(C(c3ccccn3)=O)CCC2C1 c1(CC(=O)N(C)CC2OCCN(C(CCCSC)=O)C2)ccccc1S(C)=O Cc1cnc2n1CCC(C(=O)NC1CC1CNC(=O)CN1CCCCC1)C2 C1(C(F)(F)F)(C(C2CCCOC2)=O)CC2(CC2)C1 CCC(C(=O)NC(CO)CCCCNC(c1cc(OC)no1)=O)C(F)(F)F c1(C(=O)NC2CN(C(Cc3ccc(C)cc3)=O)CC2C#N)ncnc2c1CCC2 C1(NC(C2C(C(N)=O)C2)=O)CC2CC1N(C(c1cncc(C(F)F)c1)=O)C2 N1(C(CC=C)=O)CCC2(CC1)C(OC)CC2NC(c1ccc(C2(CC)CC2)cc1)=O C(CC)(CCC(=O)OC)OC(C=C(CCC)CCC)=O c1(C(=O)OC(C)C(=O)N(C)C)cccc(C#CC2CC2)c1 S(=O)(=O)(c1ccc(C(N)=O)cc1)NC(C(c1ccc(C)s1)C)=O CC(C(=O)N(C)CC1CCC1)N(C(=O)C(C)O)C C1(C(=O)NCCNC(C(C(C)C)O)=O)CC2CCC1NC2=O c1(CC)ccc2c(CNC(N3CCN4CC5CC4(C5)C3)=O)c[nH]c2c1 C1(NC(CCc2cncc(C)c2)=O)CCN(C(=O)COCC2CCC2)CC1O Cc1c(N)ccc(C(=O)NC2(CCNC(=O)C(C)C3CC3)CCC2)c1C CCC(CCC(=O)Nc1cnn(C)c1C(N)=O)NC(=O)C(C)c1cc[nH]n1 c1(C(=O)NC23CC(CNC(C(C)SC)=O)(C2)C3)[nH]c(=N)sc1-c1ccccc1 C(=O)(C(C)(C)Cc1cccc(Cl)c1)NCC(C)CNC(=O)C(F)(F)CF c1(CN(C(=O)CCSC2CCCO2)C)sc2c(c1Br)CNC2 C12(C(=O)O)CCCC(CN(C(=O)C3CC3)C1)C2.Cc1cc2cc(n1)NC2=O N1(C(CC2CCC(NC(C3Cc4nccn4C3)=O)CC2)=O)CC2(CCC2O)C1 N1(C(C2(COC)CC2)=O)CCC(C)C(C(=O)NCc2ccc(CO)cc2)C1 c1(NC(c2n(CC(=C)C)nnn2)c2c[nH]nc2C(F)F)ccc2ccncc2c1 c1(CCNC(COCC=C)C(=O)Nc2cc(F)ccc2F)ccc(F)c(Cl)c1F c1(OC)ccc(C(=O)NCCC(C)N(C(=O)CO)C2CC2)c2ccccc12 c1(C(N2C(C)CN(C(C3CCC(=O)O3)=O)CCC2)=O)cc2n(n1)CCNC2=O c1(CC)cc(C(=O)NCC(C(C)(C)C)NC(c2cccc(F)c2)=O)ccc1OC c1(C(C)C)ccc(CNC(N2CCC(CC(=O)O)C(C)C2)=O)cc1F C1(C(=O)NCC2CN(C(CCC(C)(C)C)=O)C(C)(C)C2)COCC2(CCC2)O1 c1(C(N2CC3C(CNC(CCOC)=O)(C3)C2)=O)cc2c(nc1O)CCCC2O c1(OC)ncc(C(=O)N(CCCNC(=O)C(C)COC)C(C)C)cn1 c1(C(N2CCC3(NC(CCCCOC)=O)C(C2)C3)=O)cc2cc(F)cc(F)c2[nH]1 c1(C(N(C)CC2CCCCN2C(c2cnn(CCO)c2)=O)=O)occ2c1CCC2 N1(C(CC2N(CC)C(=O)CC2)=O)CCOCC(CNC(=O)C(C)(C)C2CCC2)C1 C(N=c1[nH]cncc1I)C1(N(C)C)CCN(C(CN(C2CCS(=O)(=O)C2)C)=O)C1 c1(C(N2C(c3ccccc3)CC(C)C2)=O)cc(N)ccc1S(C)(=O)=O c1(C(=O)NC(CNC(C(CC)N(CC)CC)=O)CO)ccc2c(cnn2C)c1 C1(C(N(C2CC2)CC2N(C(CC(C(=O)OC)C)=O)CCC2)=O)CCn2nncc2C1 c1(CC)ccc(OC)c(-c2ccnc(CC(=O)Nc3[nH]nc(Br)c3C(N)=O)c2)c1 CCC(C)C(O)C(=O)NCC12CC(NC(c3cc(C)sc3C)=O)(C1)C(C)O2 N1(C(C(C)(C)c2ccccn2)=O)CCN(CCNC(=O)Cn2cncn2)CC1 CC1CC2(CC(C(=O)NCC3CC3CNC(=O)COCc3nc[nH]n3)C2)C1 O=C1OCCCN1C(=O)C(O)C1CC1 N1(C(C(CC)Cc2cccc(C)c2)=O)CC(NC(=O)CC=C(Cl)Cl)C(C2CC2)C1 C1(NC(COCC#C)=O)CCN(C(=O)CN2CCC(C)CC2)CCC1CO N1(C(c2c(C)[nH]cc2)=O)CCC(O)C(N(C)C(C2C=CCCC2)=O)C1 CC1(C)CC2(CC(CNC(=O)OC(C)(C)C)C2)C1.C12(CCCC1)CNC(=O)N2 Cc1nn(C)c(Cl)c1C=CC(N1CC(NC(c2sc(Cl)cc2Cl)=O)C(C)C1)=O C(CCCC(=O)NC(C)CC(C)NC(c1ccccc1C(F)F)=O)OCC C1(C(N2C(CCC)COCC2)=O)CC2CC1CC2NC(=O)CC1CCCC(C)O1 c1(C(=O)NCC2CCN(C(C3(CO)CCC3)=O)C2)n[nH]c2c1CCC2 N1(C(CCCCCN(C(C2CC(C)OCC2)=O)C)=O)CC2CC(C)(C)C2C1 C1(CNC(c2ccc(SC)s2)=O)CCC2(CN(C(c3ccc(C)cc3O)=O)C2)O1 C1(CC(=O)N(CC(C)(C)CNC(c2cnc(C)nc2)=O)CC)CCC(=O)NC1=O c1(Nc2ccc(CCNC(=O)CO)cc2)ncnc2c1CNCC2 c1(CNC(C2CCC(C(=O)Nc3cc(F)cc(Br)c3)C2)=O)ncc2ccccn12 Cc1ccc(C(=O)NC2CCCCC2CNC(C2CC(=O)N(C)C2)=O)cc1 N1(C(C2(OC)CCC2)=O)CC2CCCC(CNC(=O)CC3(C)CC3)C2C1 C1(C(=O)NCC(C)N(C(=O)CCCC(=O)N(C)C)C)=CN=CC=CN=C1 N1(C(c2c(CC)cno2)=O)CCC(CF)(NC(=O)CNc2ccc(F)nc2)C1 C1(COC)CN(C(=O)CNS(=O)(=O)c2cccs2)CCN1C(C12CCCC1C2)=O C(=O)(CC(C)C(F)F)N(CCCN(C(CC)C(=O)N(CC)CC)C)CCO CC(CC(=O)NCC1CC(NC(C2CC(F)CN2C)=O)C1)C(C)(C)C Cc1cc(CC(=O)NC2CCCC(C(F)(F)F)C2)ncn1 c1(CC(=O)NCC(CC(C)C)NC(c2cccc(=O)o2)=O)cccc([N+](=O)[O-])c1 C12C(CCN1C(=O)CCSC)C(=O)NC2.c1(SCC)ncoc1C1CC1 C1(C(=O)NC2C(NC(C(n3ccc(C)n3)(C)C)=O)CCOC2)CC12CC(C)(C)C2 c1(C(N2CC(CC=C)(C(=O)O)C2)=O)ccc2nc(O)n(CC(=O)OC)c2c1 C(=O)(CCCN=c1nc2c(cnn2C)c(NC2(CN(C)C)CCC2)[nH]1)NC c1(C(=O)NC2C(NC(c3scc(C)c3C)=O)C2)ccc2cn(C)nc2c1 c1(N(C)CC2CCN(CC)CC2)nc(C)cc(=NCC2CNC(=O)C2(F)F)[nH]1 CS(=O)(=O)c1ccnc(N2CCSCC2C(=O)NCc2ccccc2S)n1 Cc1cnc(C(N2CCCC2CNC(c2cnc(C(F)(F)F)cn2)=O)=O)nc1C c1(NCCCSCC)ccc(S(=O)(=O)NC(c2ccoc2)C)cc1F c1(CC(=O)NCC(C)(CO)NC(c2cccnc2C(F)(F)F)=O)cncnc1O c1(C(N2CCC(N(CC#C)C(C3CCCO3)=O)CC2)=O)cccc(F)c1OC Cc1nc(O)nc(S)c1C(=O)NC1CCCCN(C(=O)CNc2ncccn2)C1 C(CCN=c1[nH]c(=NC2CCC(C3CC3)C2)c2ncccc2[nH]1)OCCO c1(C(=O)NC2CC3CC2N(C(c2cncs2)=O)C3)ccc2cnnc(O)c2c1 N1(C(CCCC#N)=O)CCC(C2CCN(C(C3CCCOC3)=O)CC2)CC1 C(=O)(CC(C)(C)C(=O)NCCC1CCC(NC(c2c(C)nc(C)n2O)=O)C1)OC C(=O)(CCCC(=O)N(C1C2CN(C(=O)C(F)CC(C)C)CC12)C)N(CC)CC O=C(CCC(CF)CF)NCC1(CO)CCN(C(=O)CC2CCOCC2)CC1 n1(CC)nnc(C)c1C(=O)NCC1CN(C(=O)Cn2cc(C(F)F)cn2)CC1O C(c1c(C)noc1C)=CC(=O)NCCOC1CCN(C(C2(CC)CC2)=O)CC1 C1(NC(c2cc(CCC)[nH]n2)=O)CC2(C1)CC2C(=O)N(C)CC1(C)CCC1 C1(NC(c2ccc(C(C)C)nc2O)=O)CC1C1CCCN(C(C2(CF)CC2)=O)C1 Cc1ccc(C=CC(=O)NC2CCOCC2C(=O)NC23CC(F)(C2)C3)cc1 C(C)(C)(CCC(=O)NCCC(F)=C(F)F)NC(C)=O CC(C(=O)OC(C)(C)C)C(=O)N(CCNC(=O)CC1CCCC1(F)F)C CC(CC1CCC1)C(=O)N(CCCNC(c1cc(Br)sn1)=O)C C1(C(C(=O)NC2COC2)N(CCC)CC2CCOCC2)CCOC2(CCC2)C1 Cc1cn(C)nc1C(=O)NCC=CCC(=O)NC1C2CCCOC12 C(c1ccncc1)=CC(=O)NCC#CC(=O)NC1CCC(OC)C1 c1(C(C)C)cccc(C(=O)N(C2CCN(C(C3(CF)CC3)=O)CC2)C)n1 N1(C(=O)Cc2csc(S)n2)CCC2CCN(C(=O)CSc3nncs3)C2C1 C1(CNC(c2c(CNC(CCCNC(N)=O)=O)occ2)=O)CC2CCCC2C1 O=C(C1=C(Cl)CC1)NC1C(N2CCC(OCC(=O)NCC3CC3)C2)CCC1 c1(C2(C(=O)NC3CC(N(C)C(c4ccco4)=O)C3)CCCC2)cccc(Cl)c1F CC#CCCCC(=O)N1CCN(C(=O)CC2(C=C)CC2)C2CC12 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)N(CC1N(C(c2cc(C)ns2)=O)CC1)CCO CC1=CCCN(C(c2sccc2CNC(=O)CN2C(=O)CNC2=O)=O)C1 C(=O)(C1=NNC(=O)CC1)N1CC2N(C(c3scc(C)c3)=O)C2C1 C(C(O)C(=O)OC1CC(Nc2ccsc2C)C1)=CC C(=O)(C(C)CC1CCC1)NC1CN(CC(F)F)C1.C12CC(C1)C(=O)N2CC c1(C2(C)N(C(C3CCC(C(=O)NC(C4CCCC4)C)C3)=O)CC2)ccc(F)cc1 C(=O)(C(CCC(N)=O)NC(c1ccc(OC)cc1)=O)NCC(C#C)CC1CC1 c1(NC2CCN(C(C(=O)OC)c3cnsc3)CC2)ccc(C)c(C)c1 C1(NC(c2cnc(C)s2)=O)CCCN(Cc2ccc(Cl)c(F)c2)C1C c1(C(N(CC(C)O)CCNC(C(C)OCC#C)=O)=O)cccc(OC)c1C N1(C(c2c(C)nc(CC)s2)=O)CCCC(C)C1CNC(c1cc(O)cc(O)c1)=O CC(O)C(C)(C)C(=O)NCC1CN(C)CCN1C(C1CC(C#N)C1)=O N1(C(c2n[nH]c(CC)c2F)=O)CCC2(C1)CN(C(c1c(F)cc(Cl)cc1F)=O)C2 CC1CCCC(C)N1C(c1ccc(NC(=O)CCCNC(N)=O)nc1)=O N1(C(C(CCCC)O)=O)CC2(CCCCN(C(c3cnn(CC(C)C)c3)=O)C2)C1 C1(C)(CNC(C(C)OCC(F)(F)F)=O)CCN(C(C2CC(CCO)C2)=O)C1 N1(C(CN(C(C)=O)C)=O)CCC(CNC(C2(C)C=CCC2)=O)C(F)(F)C1 N1(C(c2cn(CCC=C)nn2)=O)C2CCC1CN(C(c1ccc(C#N)s1)=O)CC2 C1(NCCC23CC(n4cc(C(C5CC5)COC)nn4)C2C3)CC2CS(=O)(=O)CC2C1 N1(C(Cc2scc(C)c2)=O)CCC2CN(C(=O)C(C)(C)c3cscc3Cl)CCC12 N1(C(CCC2CCC(NC(C3C(C(C)(C)C)C3)=O)C2)=O)CC2CC2(CO)C1 C1(NC(C)C2CC2)CC(NC(C)CC2CC2)C1n1cccn1 C1(C(=O)NCc2c(C)n[nH]c2)CC(O)CN1C(C1CCCN1C)=O C(=O)(CCCC(C)=O)Nc1c(Nc2ccc(N(C(C=C)=O)C)nc2)n[nH]c1 C1(CC(=O)NC2CC(O)C2)CCCCN1c1ncccn1.C12CCCN(C1)C2=O c1(C(=O)NCC2C3CN(C(c4c(C)cccc4)=O)CC32)cnc(O)c(F)c1 C1(CNC(c2c(C)sc(O)n2)=O)CC(C)CCN1C(=O)C=CC1CCCO1 N1(C(c2c(C)ccc(SC)c2)=O)CC(C)N(C(c2c[nH]c(=N)cc2C)=O)CC1C Cc1cc(=N)[nH]cc1C(N1CCC(NC(=O)CC2CC3CCC2CC3)C1(C)C)=O C1(OC)CC(C(=O)NCC2(C3CC3)CC2)N(C(=O)Cc2cnccn2)C1 N1(C(C2N(C(C(C(C)(C)C)=O)=O)CSC2)=O)CC2CN(C)CC2(C)C1 c1(NC(C2C(Nc3c(C)cncn3)C2)=O)cc(F)cc(I)c1 N1(C(c2nccc(OC)c2)=O)C2CC1CN(C(=O)Nc1ccc(OC)cc1)C2 n1(C(C(=O)NCCCN(C(=O)CC2CCC3CC23)CC)C)ccnc1C(C)C N1(C(CCOC)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C2CCCCC12 C1(CNC(=O)NC(C2CCCN2CCC(C)C)CC)CC2CC1C2 c1(C(N2C(C(N(CC(CC)NC(C)=O)C)=O)CCC2)=O)cc2c(O)cccc2[nH]1 C1(NC(C2(CCOC)CCC2)=O)CC(O)CN(C(c2coc(Br)n2)=O)C1 c1(CN2CCC(NC(COC)=O)C(OC)C2)ccc(C#CCO)s1 N1(C(c2cc(C)n(C(C)C3CC3)n2)=O)CCC(CNC(C2CCCO2)=O)C(C)C1 Cc1cccc(C(=O)NC(CC2CC2)C(=O)N(C2CCNC2=O)C)c1O Cn1ccc(C(N2CCCC(C)(C(N3CCC(CCF)C3)=O)C2)=O)cc1=O c1(C(C)C(=O)OC(CC(C)(C)C)C(F)F)ccc([N+](=O)[O-])cc1F C1(C(C)C)C(=O)N1.C1(C(=O)NC(C2CCCCC2)C(C)C)CCCCC1 C(=O)(CCS(C)(=O)=O)N1CCC(O)(CN(C(C(C)C(F)F)=O)C)C1 Cc1c(C(=O)NCCC(C)(C)NC(C2CC2C(F)(F)F)=O)ccn1C(C)C C1(CC=C)CC(O)CC(CNC(=O)C(C2CC2)NC(=O)CC)O1 N1(C(C=CCCC)=O)CC2C(NC(c3cc(C)n(CC)n3)=O)C2C1 C1(C(N2C(C)CN(C(=O)COC3CCCC3)CC2)=O)CC(=O)c2ccccc2C1 c1(CCC(N2CCC(N(C(=O)C(F)C3CC3)CC)C2)=O)cc(C)sc1C N1(C(CC(C)NC(C(C(C)O)(F)F)=O)=O)CC2(CCOCC2)C1 Cc1cccc(OCCCOC(C2C(O)C(O)CN2C(=O)OC(C)(C)C)=O)c1C N1(C(c2n(CC)c(O)nc2)=O)CCC(C)C(N(C)C(c2ccc(OC)nc2)=O)C1 CN1CCN(C(=O)CC2CCCO2)C(CNC(c2cnn3c2OCC3)=O)C1 Cc1cccc(N(C(=O)C(C(C)C)C2CC2)C)c1.C(C(O)C)NS(C)(=O)=O N1(C(C2(C(=O)OCC)CCC2)=O)CC2(CCN2C(=O)CC2CCCSC2)C1 c1(C(=O)NC2CC(N(C(C3(OC)CCCC3)=O)C)C2)cc(S(C)(=O)=O)oc1C C1(C(N2CC(C)C(O)C2)=O)CCNC12CCOCC2 C12(C(N)=O)CC1CN(C(c1ccnc(O)c1)=O)C2.c12occc1CNC2=O N1(C(CN(CCOC)C)=O)CCOC2(CCCN(C(C3CCC(=O)NC3)=O)C2)C1 n1(C(C)C)ccc(=NC(=O)C2C3CC(O)C(C3)N2C(C2(O)CCC2)=O)[nH]1 CC(C(C)(C)CO)NC(=O)C(C)(C)C1CCN(C(C2CCCC2F)=O)C1 c1(CNC(C2(Cl)C(C(C)=O)C2)=O)ccc(C(=O)N(C)CCN2CCCC2)nc1 Cc1ccc(-c2cccc(C(C(=O)N)N(C)C)c2)cc1.C(C)(C)(C)OCC1CC1 CN1CCC(C)(C(N2CCOC(CNC(c3cnn(CCF)c3)=O)C2)=O)C1=O c1(C(N2CC3(CN(C(c4c(C)cco4)=O)C3)C2)=O)ccc2cccnc2c1 C1(NC(C(C)Cn2cccc2)=O)CCC(C(=O)N(C2CCOC2)CCO)CC1 c1(C(N2CCN(C)CC2CN2CCC(N3CCC3)CC2)=O)cc(Cl)c(Br)c(Cl)c1 N1(c2nccc(OC)n2)CCCC(C)(C)C1CNC(=O)CC1CC2CCC1CC2 c1(C(=O)NCCN(C(=O)CP(C)(C)=O)CCOC)nc2n(c1Cl)CCCC2 C(C)(CNC(=O)Cn1cc(C2CC2)nn1)(C(C)C)NC(c1ccc(C(C)C)o1)=O c1(C(N2CCOCC(F)(CNC(C(C)=CC)=O)C2)=O)ccc2cnnc(O)c2c1 C(=O)(C1CCCc2cc(O)ccc21)NC(C)CCNC(=O)CSc1nncs1 c1(OC)ncccc1C(=O)N(C1CCN(Cc2nncc(-c3nn[nH]n3)c2)C1)C c1(C(=O)NCC2CN(C(CC3C(C)=NOC3=O)=O)C2)c(C)nn2ccccc12 N1(C(C2(COC)CC2)=O)CCC2(CNC(c3sc(OC)nc3C)=O)CCCCC12 c1(C(=O)N(C(C)(C)C)Cc2cccc(OCC)c2)cnc2sc(Br)cn12 c1(CN2C(C(=O)Nc3cn(COC)nc3)CC2)cc2ccccc2nc1OCC C1(C(=O)NCC(=C)F)(CC)CCCN1C(=O)CC1CCC1 N1(C(c2c(C(C)C)nns2)=O)CC2C(CNC(c3c[nH]c(Br)c3)=O)C2C1 c1(C(N2CC(CNC(=O)CCc3cncs3)C(F)(F)C2)=O)ccc2nncn2c1 CCC1=NOC(C(=O)NC(C)(CSC)C(=O)NCC2(COC)CC2)C1 c1(C(N(C(C)C)CCNC(c2cc(C(F)F)n(C)n2)=O)=O)cnc2n1CCC2 Cc1c(C(=O)N(C)CCOCCCNC(=O)C(C)C(C)O)sc2ccc(F)cc12 c1(OC)ccc2c(C(=O)NCCN(C(=O)Cc3sccc3C)C3CC3)c[nH]c2c1 c1(C(N2CC(C)C(CCNC(=O)OC(C)(C)C)C2)=O)ccnc2[nH]c(O)nc12 CC(C)(CCCNC(C1CN(C(N)=O)C1)=O)NC(=O)CC1CCC(O)C1 c1(C(=O)NC(C2CN(C(=O)COC3(C)CCC3)CCO2)C)ccc2nnnn2c1 N1(C(C2C(CC)CCC2)=O)CCN2CCN(C(=O)C(C)(C)CS(C)(=O)=O)CC2C1 C1(C)(C(=O)NCCN(C(C(C)=C2CCC2)=O)CC2CC2)C=CCC1 n1(CC)cc(Br)c(CN(CC(C)(C)[N+](=O)[O-])C=O)n1.N(C)CC C1(C(=O)NCc2c(CC)nns2)C(C2CC2)CCN1C(c1ncn(C(C)C)n1)=O CC1CN(C(=O)CCc2ncco2)CC1NC(C1(n2cccn2)CCC1)=O C1(CN(C(=O)CCOc2ccccc2C(C)=O)CC)CCN(C(=O)C2CC2)CC1 C#Cc1cnn(CC(N2CCC(C(C)(C)NC(=O)C=CCN(CC)CC)C2)=O)c1 C1(OC)CC(C(=O)Nc2ccn(C)c2)N(C(=O)C(C(C)C)C2CCC2)C1 C1(C(C)NC(=O)CSc2nc[nH]n2)CCN(C(C2(CO)CCCCC2)=O)CC1 C1(CNC(C2CC3(CCC3)CO2)=O)CC12CCN(C(c1ccnnc1S)=O)CC2 Cc1ccc2c(c1)CC(C(=O)NCC1CC(NC(=O)Cc3ccc(F)cn3)C1)S2 C(CCC(O)C(=O)NC1CCCCC1CO)NC(c1cn(C(C)C)nn1)=O N1(C(C(C2CN(C(CCC(N)=O)=O)C2)O)=O)CC2CCCC(O)C2C1 C=C=CCCC(=O)NC1(CC=CC(N2CCN(CC(C)O)CC2)=O)CCC1 CN1CC(C(=O)NC(C)(C)C=CC(=O)NC2CCC(=O)N(C)C2)CCC1=O c1(CC(=O)NCCC2(C(=O)OC(C)(C)C)CCC2)cccc2c1OCO2 c1(C(=O)NCC2(O)CCN(C(c3cc(C)no3)=O)CC2)cc(Br)c(C)cc1O C1(NC(C2C(=C)C2)=O)(CO)CCN(C(c2c(C)coc2-c2ccccc2)=O)C1 C1(NC(c2c(C#C)c[nH]n2)=O)CCC(C)N(C(c2cnn(CCO)c2)=O)C1 C1(=O)CC(CNC(=O)OCC)O1.C1(Cl)(C(c2ccccc2)OC)CC1(F)F c1(C(N2C(C(=O)NC3CONC3=O)CC(C)C2)=O)ccc2c(c1)OCO2 C1(NC(c2cc(C)nnc2)=O)CCC2(CCN(C(c3onc(C)c3C)=O)CC2)C1 C(=O)(CC(C)(C)C(=O)OC)NC(C(=O)N(CCC)CCN(C)C)Cc1ccoc1 N1(C(CC(C)(C)C#N)=O)CCC2(CCOCC2)C(CNC(c2ccc[nH]2)=O)C1 N1(C(CNC(C)=O)=O)CCC(NCCNC(=O)CNC(c2ccncc2)=O)C1.N C(C(=O)NCC12CC(NC(=O)CC3SC(=N)NC3=O)(CO1)C2)(C(C)C)SCC CC1CN(C(=O)C=CSc2nc[nH]n2)CCN(C(=O)CC2(N(C)C)CCCC2)C1 C1(NC(CCCc2nc(C)sc2)=O)CC(C)CN(C(C2(C(C)C)CC2)=O)C1 c1(C(=O)NC(CN(C(C(C(C)C)NC(N)=O)=O)C)C)cc(F)cnc1O N1(C(CCCC=C)=O)CCC(C2(NC(c3cccc(=O)n3C)=O)CC2)C1 C(=O)(C1COc2ccccc21)NCc1cccc(NC(C(C(C)C)O)=O)c1 C1(NC(C2CC(F)(F)C2)=O)C2CC3CN(C(=O)CC4CN5CCN4CC5)C1C3C2 C12(C(N3CC=CC(NC(c4n(CC)cnn4)=O)C3)=O)CCCC1C2(F)F C1(C(=O)NC(COC)C2CC2)CC(C)(C)CN1C(c1cccc(=O)n1C)=O C(CCCCCNC(C12CC1CCN2C(c1[nH]ccc1C)=O)=O)OC c1(CC(=O)N(CC(C)NC(=O)CN(C)C)CC)c[nH]c2ccc([N+](=O)[O-])cc12 c1(NCC(C(C)(C)C)NC(c2scc(C)c2)=O)nc(Cl)nc(C)c1F N1(C(CCCOC(C)(C)C)=O)CC=CC(NC(C2(CS(C)(=O)=O)CCC2)=O)C1 CC1CC(C(=O)NCCCCC(CO)NC(C2(C)CC=CC2)=O)CC(C)(C)C1 C1(NC(C2(CCOC)CCC2)=O)C(C)(C)CN(C(=O)C(C)N2CCC2)CC1(C)C c1(C(C(=O)NN(CCOCCOCC)CC)OCOC2CCCOC2)occc1Br C1(NC(c2csc(Cl)n2)=O)CC2CC1N(C(=O)CC1CCOC1=O)C2 c1(CC)onc(C)c1C(=O)NCC1(OC)CN(C(C2CN(C(N)=O)C2)=O)C1 C=CCCC(C(=O)NC1CCCN(C(=O)CCSCC#N)CC1)c1ccccc1 C1(OC)CN(C(C2CC2(C)C(F)F)=O)CC1C(=O)NCc1nccc(C)n1 C1(C(=O)NC2C3CN(C(CNC(=O)OC)=O)CC2C3)CC2C(C1)C2(C)C N1(C(CN(C)C)=O)CC(O)(CCNC(C2CCN2S(C)(=O)=O)=O)C1 CC1(C)CCC2(CC1)CN(C(NC1CCc3ccccc31)=O)CCO2 c1(CC(C)C(=O)NCCCNC(C2CC2c2cccs2)=O)cccc(Br)c1 N1(C(CCS(=O)(=O)NC)=O)CC(NC(c2scc3c2OCCO3)=O)CC12CCC2 CC(C)C(O)C(=O)NC1CCCC(NC(c2sccc2C2CC2)=O)C1 N1(C(c2c(C)nsc2C)=O)CC(N(C(=O)CCn2cccc2)C)C2(CC2)C1 N1(C(C2(N(C)C)CC2)=O)CCC2CN(C(c3ccnc(C4CC4)n3)=O)CC12 CC(C)(C)CCCC(=O)N1CC2CCN(C(=O)CCCCOC(C)(C)C)C2C1 c1(NC(C(c2nc(C)c(C)o2)N(CC(F)F)CC)=O)cccc(OC)c1 C1(OC)CCC(C(N2CC=CC(NC(=O)CC3CC3C(F)(F)F)C2)=O)CC1 C1(OCC(=O)NCC(c2ccccc2F)F)CCC(F)(F)CC1 CCC(C#N)C(=O)N1CCCC1c1cccc(-c2ccccc2)c1 C1(OC)(CNC(C2(C)CCC(=O)N2)=O)CCN(C(C2CCC2C#N)=O)C1 c1(C(=O)NCCCOC)c(F)cc(S(=O)(=O)N=c2nnn(C)[nH]2)cc1F C1(CCC)CN(C(c2ccc(N)c(F)n2)=O)CCN1C(=O)CCc1ncccn1 C1(C(N(CC(C)OCC)C)=O)C2CC3C(C2NC(c2c(CC)cnn2C)=O)C13 N1(C(C=CCNC(C(CO)OC)=O)=O)CCC(O)C1C c1(-c2ncc(CN(C3CCC4(CC3)CC4N)C)s2)ccc2c(c1)OC(F)(F)O2 c1(NC(N2CCC(C3CCCN3)C2)=O)cn(C2CCOC2)nn1 c1(CNC(CC(C)N(C)C)=O)n[nH]c2c1CN(C(=O)CN=S(C)(C)=O)CC2 c1(NC(N2C(NC(=O)CCCc3cccs3)CCC2)=O)ccc(C(F)(F)F)cc1 c1(C(N(C(CNC(C(CC)SC)=O)C2CC2)C)=O)cc(CO)oc1C C(C(C)C)(C(O)C(=O)NCC1CCCCN(C(c2nc(=N)cc[nH]2)=O)C1)OC c1(CN2CCC(CC(=O)NCC3CCC4(CC3)CC4)C2)cccc(O)c1Br C1(N(C(C2CCCN2C)=O)CC)CCN(C(=O)OC(C)(C)C)CC1 c1(C(C)(C)C)cccc(N2CCCCC2)c1.C1CC(F)(F)COC1=O N1(C(C(C(C)C)=O)=O)CCN(C)CC1C(N1C(C)CCC1(C)C)=O CCCCCCCCC(C)C(=O)NCCCC1(NC(C2CC2C(N)=O)=O)CC1 c1(C(=O)NC(CNC(c2nc(CC(C)C)sc2)=O)CO)ccc(Cl)c(NC(C)=O)c1 N1(C(CSCCN(C)C)=O)CCCC(N(CCF)C(c2ccnn2CC#N)=O)C1 C(=O)(CCCCCF)NCc1c(C(=O)NC(c2cccnc2F)C)cco1 C(C)(CC(=O)NCC1(CNC(c2c[nH]nc2C2CC2)=O)CC1)(C(F)(F)F)N(C)C C=CCC(C)C(=O)NCc1oc(C(=O)NCCC(CC)CO)cc1C Cc1c(N)ccc(C(=O)NC2CCN(C(C3CCCC3(C)C)=O)C2)c1Cl C(CC(C(=O)NC1CC1(C)C(C)C)NC(C12CC(CO)(C1)C2)=O)=CC C1(NC(C(CC2CCC2)OC)=O)CCN(c2nnco2)CC1O c1(OC)ccc(C(CNC(=O)CC2CC3CC3C2)NC(C2(Cl)CC2)=O)cc1 n1(CC(=O)NC2CC(CO)N(C(=O)CCCCN(C)C)C2)ccc2ccccc12 CCCCCCC(CC)C(=O)NC1CCC2CN(C(=O)C(C)(C)F)CC2C1 c1(C(=O)NC(C)CNC(C2CC2C(=O)OC(C)(C)C)=O)cc(Br)c2n[nH]cc2c1 c1(CC)cc(C(=O)NCC2CN(C)CCN2C(=O)Cc2nc(=N)[nH][nH]2)cc(F)c1 Cc1noc(C(=O)NCC2CC(NC(=O)C(C)C#N)C2)c1C.c12ccc(s1)C2=O CC1=CCN(CC(=O)N(n2cc(CCc3cccs3)nn2)C)CC1 O=C1CNc2cc(NC(=O)CC3(c4ccccc4)CC3)cnc2N1 C(CO)(CCCCNC(C1(C(N)=O)CC1)=O)NC(C1(C)CCCCO1)=O C1(NC(C(CC)=CC)=O)CCC2CCN(C(C3CC3F)=O)C12 C(CCC)(C(=O)NC(C)C(C)NC(=O)C(C)NC(=O)CC)=CCC c1(C(=O)NC(C2CC=CCC2)c2ccccc2)cnn2cnnc2c1 CC1CCC(O)(CNC(=O)C(Cc2ccoc2)NC(c2cc(Cl)cn2C)=O)C1 CN1C2CCC1CC(=CC(N1CCC(NC(=O)C3CC3)C(O)C1)=O)C2 CCCC(CC)C(=O)NCCCN(C(=O)CC(C(F)(F)F)n1cccn1)C c1(NC(c2ncc(Cl)cn2)C)ccc(S(=O)(=O)NCC2(N(C)C)CC2)c(Cl)c1 c1(N2CC(O)(CCNC(c3nn(C)c(C(N)=O)c3)=O)C2)ncnc2scnc12 C12(NC(c3cnn(CC)c3C)=O)CCC(CNC(=O)Cc3ccno3)(C1)OC2 c1(C(COC(CC2CN(C(C)=O)CC(C)C2)=O)=O)ccc([N+](=O)[O-])cc1 N1(C(CCC(=O)OCC)=O)CC2(CCC(N(C(C(=O)N(C)CC)C)CC)C2)C1 c1(-c2nc(C(C)C)sc2)n[nH]c2ccc(C(=O)Nc3cccc([N+](=O)[O-])c3)cc12 c1(-c2c(C)occ2)nc(C(c2nncn2C)C)n(CCC(C)(C)C)n1 C1(C(=O)NC(C)C(=O)NCCCCC(=O)NC2CCC(=O)N2)CCC(C)(C)CO1 c1(C(=O)NCC2(O)CCN(C(C3(C(CC)(F)F)CC3)=O)CC2)ccc2cnoc2c1 CC(C)C(C)C(C)CC(=O)N1CCCCC1CNc1nc(O)c2c(ncn2C)n1 c1(C(N2CCCCC(CNC(C(C(C)(C)O)F)=O)C2)=O)cccc2sccc12 C(=O)(CCCC(C)(F)F)N(C)CC1(O)CCN(C(=O)CC2CCC(O)C2)CC1 n1(CC(N2CCC(N(C(c3c(C)csc3)=O)C)C2)=O)nc2c(n1)CCCC2 C1(C(N(CC(CNC(c2c(OCC)nccc2)=O)C)C)=O)CN2CCN1CC2C c1(C(N2C(CNC(c3ccc4c(c3)CC4)=O)COCC2)=O)ccc([N+](=O)[O-])[nH]1 C12(C(=O)NCC(C(=O)NCCN(CCO)CC)N(C)C)CCCC1C2(F)F C12CCN(CCC1CO)C(=O)C=CC(=O)N2.c1(C(C)=O)cnc2c(ccn2C)c1 C(CCCC(=O)NC1CCOC1C(N1CCC(CCCO)CC1)=O)OC C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC2(CN(C(=O)CC3CC(O)C3)C2)C1 C(CN=c1[nH]cc(C#N)cc1C)N1CCN(C(CCS(CCCC)(=O)=O)=O)CC1 C(=O)(C(C(=O)OCC)C(C)C)NC(CC)CNC(=O)CCc1cnc(C)o1 CC(CC(F)(F)F)C(=O)NCC1CCCN(C(=O)C=C2CCCCC2(C)C)C1 N1(C(=O)COCCOCCO)CC2CC(C1)N2C(C12CC1CNC2=O)=O c1(OC)ccc(CC(O)C(=O)Nc2cccc(NC(C3(CO)CCC3)=O)c2)cc1 C#CC1(C(=O)Nc2cnn(CC(C)C)c2)CCN(C(C2C3CCC(F)(F)C23)=O)C1 CCC(C)(C)C(O)C(=O)N(C1CCC(NC(=O)C2=CCCO2)CC1)C c1(CNC(C(N2CC(C#C)NCC2)=O)=O)nn(C)c(C)c1S(N)(=O)=O N1(C(c2c(C)oc(Cl)n2)=O)CCC2CCN(C(=O)C=Cc3cccs3)C2C1 c1(OC)cc(F)cc(C(=O)NCC2(C(N)=O)CN(C(C3(C(F)F)CC3)=O)C2)c1N C(=O)(C(C)S(=O)(=O)C(C)C)N1C2(CNC(Cc3c(C)cccn3)=O)CC(C1)C2 C(=O)(CC(C)CC(F)(F)F)NCc1cncc(NC(C)=O)c1 C(=O)(CC(C)CCC=C(C)C)NC1CN(C(c2nc(CC)oc2C)=O)CC12CC2 C(C(O)C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1(CF)CC1)=CC n1(NC(C(Cc2ccsc2)NC=O)=O)cc([N+](=O)[O-])cn1 N1(C(C=CCCOC)=O)CC(CNc2ncc(C(F)(F)F)cc2OC)OC(C)(C)C1 Cc1noc(CCC(=O)NCC2CC(F)(CNC(C3(CC#N)COC3)=O)C2)n1 CCC(O)C(C)C(=O)N1CCN(CCNC(=O)C(c2cc(Cl)cc(Cl)c2)O)CC1 C1(C(=O)NC)CCN(C(=O)C(CNC(C2CCC(O)CC2)=O)N(C)C)C1C c1(SC)nc(NC(C2CC23CC(O)C3)=O)cc(N2CC(CC(C)OC)C2)n1.C(F)F Cc1cc(C(=O)NC(C(=O)NC2(CO)CC3(CCC3)C2)C2CCCC2)c(C)cn1 C(C)(N=c1nc2c(ncn2C(C)C)c(NCC2(C)CCC2)[nH]1)c1cc(C)on1 C1(CNC(c2cc(C)sc2)=O)CN(C(=O)C(CC(C)C)NC(N)=O)CC12CC2 CCC(C)C(=O)C(=O)NCc1cncc(C(=O)NCCSC(C)(C)C)c1 c1(CC)cnc2ccccc2c1C(=O)NCCC1CN(C(=O)CS)C1.C(C)(C)(C)S CC1Cc2c(C(=O)OCc3ncccc3Cl)cccc2CO1 C(=O)(C(O)CC(N)=O)N1CC(CCC)C(NC(C2CCCC23CCC3)=O)C1 Cc1cn(C)cc1C(=O)NC1(CNC(C2(C)CC2Br)=O)CCCC1 N1(C(c2c(CC)onc2C)=O)CC=C(C(=O)N(C2CCC2)C)CC1 c1(C(N2C(CNC(c3cc(Cl)nnc3Cl)=O)CCC2)=O)cc2ccncc2[nH]1 Cc1ccc(F)c(C(=O)NC2CCCC(N)CC2)c1Cl C=Cc1cncc(C(=O)NCC=CC(N2CCC(CC(N)=O)C2)=O)c1 Cc1ccc(-c2cc(OCC(N3CCC(CO)C3)=O)n(C)n2)cc1 CCC(C)CCCC(=O)N1CC(O)CC1(C)C(=O)NCc1cnc(C)o1 C(=O)(CCP(C)(C)=O)N1CC(CCCNC(CN(CCC)C)=O)OCC1 N1(C(C2(C)CC2)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC1c1ccc(F)cc1 C1(NC(C(C)S)=O)CC2(C1)CC(NC(C1(c3ccccc3)CC1)=O)C2 CCC(C)C(C(=O)NC1(C(=O)NC(C)(C)CCCO)CCSC1)N(C)C CC1(C)CC(COC(c2sccc2C2CC2)=O)CO1 c1(COC)ccc(C(=O)NC(C2CCCN2C(=O)CC2CCC2)(C)C)cc1F N12CC3OCCN(C3C1)C2=O.CCC1CN1.S(C)(=O)(=O)N(C(C)C)C(C)C N1(C(CCSC)=O)CCC(C(F)(F)F)C(NC(=O)CCCc2cccnc2)C1 c1(NC(C)=O)ccc(CN2CC(OC#N)CC2C(N2CCCC2)=O)cc1 C1(NC(CC)=O)CCOC2(CCN(C(c3cccc(C(F)F)c3F)=O)CC2)C1 C1(C(N(CCSC)CC)=O)C=CCN(C(C2CC(=O)CCO2)=O)C1 c1(C(N2CCCN(C(c3nc(C)n(C)n3)=O)CC2C)=O)c2c(nn1C)CCOC2 C1(COC)(NC(=O)CSCCOC)CN(C(C23CCCC2C3)=O)C1 C1(NC(=O)COCC2CC2)CCC2CN(C(c3ccc(O)nn3)=O)CCC2C1 N1(C(c2ccccc2Cl)=O)CCC=C(C(=O)N2C(CO)CCC2CO)C1 CCC(C)(CNC(=O)CCN(C)C)C(=O)NCCN(CC(F)F)C C1(C(C(=O)NCC(C)CN(C)C(C2CCCCN2C)=O)F)CCCCCC1 c1(C(=O)NCC(N(C(C(C=CC)O)=O)C)C2CC2)cccc(C)c1Cl C1(CC=C)(C(=O)N(CCOCC(C)O)C(C)C)CN(C(=O)CC2CCCOC2)C1 C1(F)(C(=O)NC2(C)CC=CCC2)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 C1(F)(CNC(Cc2cc(C)nn2C)=O)CC(N=c2[nH]nco2)C1 C(=O)(C1Cc2c(Cl)cccc21)NC1(CCNC(CC2C(C)(C)CCCC2)=O)CC1 C1(C(=O)NC2CC(N(C(C(C(C)(F)F)(C)C)=O)C)C2)CCC(S(C)(=O)=O)CC1 C(c1ccccc1F)=CC(=O)NCC1(NC(C2NC(=O)OCC2)=O)CCC1 C1(N(C(=O)CCn2nc(C)cc2C)CC)CCCN(C(=O)C#CC2(C)CC2)CC1 C(CN=c1cc(NCC2=CCCC2)nc[nH]1)c1nc(CC(=O)NCCCF)sc1 C1(CNC(=O)NCC2CCCC(F)(F)C2)CC2(COCCO2)C1 Cc1cc(C(N2CC=CC(NC(=O)CC3CC3)C2)=O)c(C)n1-c1ccccc1F N12CCN(CC1CC)C(=O)C1CC1C2=O.C1(C(=O)OCC)CC(CF)C1 C1(C(=O)NCCCOCC#C)CC2(CCC2)CN1C(=O)C(C(C)CC)N(C)C c1(C2C(C(N(C(c3ccncc3)C(=O)OC)C)=O)C2)ccc(C#N)cc1 C1(CCOC)(NC(=O)CC2(O)CCCC2)CCN(C(c2ccc(CO)o2)=O)C1 CC1(C)CCCC(O)(C(N2CCC(N(C(=O)C3=COCCC3)CCO)CC2)=O)C1 Cc1nc2cc(C(=O)NC3CCCCC3NC(C3CCO3)=O)ccc2o1 c1(NC(c2sc(Cl)cc2Cl)=O)ccc(Cl)cc1[N+](=O)[O-].CC1CN1C Cc1cccc(C)c1C(O)C(=O)N(CCNC(c1nc(C)c(C)[nH]1)=O)C1CC1 c1(CC(=O)NCC(=O)NCC(C)(C)OCCO)c[nH]c(=N)nc1O.c1(O)cnccn1 c1(C(=O)NNC(=O)N2CCNC(=O)C2)ccc(Cl)cc1Cl.C1(C(=O)O)(C=O)CCOC1 N1(c2ccc(-c3c(F)ccc(COC)c3)cn2)CCC(S(C)(=O)=O)CC1 CN1CCCN(C(=O)CCOCCCNC(c2cc(O)cc(=O)o2)=O)CCC1 C1(CN(C(C=COCC)=O)Cc2ccccn2)CC2(CCC2)CO1 C1(C(C)NC(c2scnc2C2CC2)=O)CCCN(C(=O)CCC=CBr)C1 Cc1cc(C(=O)NCCCC(C)NC(C2(CF)CCC2)=O)cc(C)c1Cl C(=O)(CCCCCC(C)C)N1CC2CCC(NC(Cc3ccc(C)cc3)=O)(C1)C2 C12(C(=O)Nc3cc(C)ns3)CCCC1CN(C(c1ccc(O)nc1)=O)C2 Cc1ccc(Br)c(CC(=O)N(C)CCNC(c2cocn2)=O)c1 C(CCCC(=O)N1CC(C(=O)NC2C=CCCC2)C(C)C1)OC c1(C(=O)NC(C(=O)NCC(=C)C)C2(O)CCC2)nn(C)cc1Cl Cn1cnc2sc(C(=O)NCCCCCCNC(C3CCCN3N=O)=O)cc12 c1(C(=O)NC2CN(C(c3cnc(OC)c(Cl)c3)=O)C3C2C3)n[nH]c2c1CCCC2 C12CN(CCC1F)C(=O)O2.CCC(CC(=O)Nc1ccc(Cl)cc1)C1CCC1 C1(C(N2CCCCC(N(C)C(c3cccn3C)=O)C2)=O)CC2CCCC(C1)C2 C(C(C)C)(C(O)C(=O)N1CCCCC(C(=O)NC(C)CC(C)C(F)F)C1)OC CC(=O)C(C)CC(C)C(=O)N(CC(C)(C)C(N1CC2CCC(CC2)C1)=O)C C1(NC(C(Cc2ncn(C)c2)O)=O)CCN(C(C2(F)CCCCC2)=O)CC(O)C1 C1(NC(CCc2cncc(C)c2)=O)CCCCN(C(c2cn(C)nc2Cl)=O)C1 C1(C(N(C)Cc2ncc(C)o2)=O)CCC(CNC(C2COC(C)C2)=O)CC1 c1(CN(C(=O)C(C)(O)CO)CCCN(C)C)ccc(Cl)c(Cl)c1 N12CCC(CC1)NCCC1N(CCC1)C2=O.C1(C(=O)OC)CCC(=O)N1 C1(C)(C(=O)NCC2CCC(C)O2)CCN(C(=O)CC2CC(F)(F)C2)C1 N1(c2cc(C(=O)OC)cc(C(F)F)n2)CC2(CC=CC2)C1C(C)C c1(CCC(=O)NC(C)CCCCNC(=O)CCC2CC2(C)C)ccc(Cl)c(F)c1 O=[N+]([O-])c1cc(NCc2ccc3c(c2)CCCC3)cc(Br)c1 c1(C(=O)NC2CCN(C(C(C)OCCCC)=O)C(C)C2)cccc2c1ncn2C C(c1cc2ccccc2o1)=CC(N1CC(C)N(C(C2(C)CCCOC2)=O)CC1)=O Cc1ccc(C=CC(N2CCC2CNC(=O)CN2CCC(C)(O)C2)=O)o1 C1(C)(CNC(C2CCN(CCC#C)CC2)=O)CCN(C(C2CCCS2)=O)CC1 c1(C(C)(C)C)nc(C(=O)NC2CC(CCNC(C3CCCS3)=O)C2)co1 c1(C(=O)NC(CNC(c2c(CC)noc2C)=O)CC(C)C)cccc2sncc12 N1(C(c2nccs2)C(=O)NC)CC(C(=O)OC(C)(C)C)C(C(N)=O)C1 N1(C(c2c(OC(C)C)cccn2)=O)CC2(CCCC2NC(C2CC2(F)F)=O)C1 N1(C(c2ccccc2-n2cc(Br)cn2)C(=O)NC)CCCC(CSC)CC1 C1(C(N(CC(CC)(CC)NC(=O)C=CC2CCOC2)CC)=O)CCc2nccn2C1 C1(NC(CCN(CC)CC)=O)CCC(NC(=O)Cn2cc(CCC(C)O)nn2)C1 N1(CC(=O)NCC2CC(C)N(c3nnc(O)nc3O)C2)C(=O)CN(C)C1=O C1(C(=O)NCC2(OC)CN(C(c3nnccc3C)=O)C2)CC2(C)CCC1(C)O2 C=CC1(CC(N2CC(O)(CNC(=O)C(C)=CCC)C2)=O)CCCCC1 C(=O)(CC1OCc2ncccc21)NCC1(C)CCN(C(c2cc(CO)on2)=O)C1 C12(NC(c3cnc(CNC(C4(C)N(C)CCC4)=O)nc3)=O)CCC(O)(CC1)CC2 c1(C(=O)NCC2N(C(C3C(OC)C3)=O)CCCC2)ccc(-c2cccs2)nc1C n1(C(CC)C)nc(CN(C)CCN2CCCCC2)nc1C1COC(C)C1 c1(C(C(=O)NCCC2(NC(CC3(C)CCOC3)=O)CCC2)(C)C)ccc(O)cc1 C(=O)(C1=CCCCCC1)N1C(CNC(=O)COCc2nc(C)no2)CC(OC)C1 c1(C(=O)NC2CN(C(c3cccc(SCCC)c3)=O)C2)cn(C)c(=O)n1C c1(C(=O)NC2CC(NC(C3(Cc4ccccc4)CC3)=O)C2)cc(Cl)c(Cl)[nH]1 N1(C(C(C)(C)CO)=O)CC2(CC(NC(=O)C3=CC(O)CCOC3)c3nccn32)C1 N1(C(C(C2CCC2)OC)=O)CCCC2(CCN(C(C3(C)CC4CC4C3)=O)CC2)C1 c1(C(N2CC(CNC(C3CC(CN(C)C)C3)=O)OCC2)=O)cc2cccnn2c1 c1(CC)ccc(F)cc1NC(=O)C(C)(C1CC1)N(C(=O)Cc1cncnc1)C C(=O)(C(CC(C)C)N)C(CNCC#CCNC(c1cc(OCC)ncc1)=O)=O.OC C1(NC(COCC(=C)C)=O)CC2CCC1N2C(=O)CCc1nnc(C2CC2)o1 Cc1nc2c(s1)CCCC2C(=O)NCC(C)(C1CCC1)NC(c1ncoc1C)=O CCCCCC(=O)NCC1CCC(N(C(=O)C(c2cccc(F)c2)(C)O)C)CC1 C1(NC(C)=O)CCC(C(=O)NC(c2ccsn2)=O)CC1.c12cccc(c1)CCN2 C(C(CC)C(C)(F)F)N(C1CCOCC1)C(c1ccc(C#C)o1)=O N#Cc1ccc2c(c1)CCCN2Cc1ccncc1-c1ccc(F)nc1 c1(NCC(C(c2nnnn2CC2CC2)OC(C)C)(C)C)nc2c(s1)CCCCC2 N1(CC(=O)NC(C(=O)N(C)Cc2cnco2)c2ccco2)CCC(C)C1 C(C)(C(C)C(=O)NCC1(SC)CCC1)NC(C1(C(C)(C)OCC)CC1)=O c1(C(=O)NC2CN(C(C3C(CCC)CCC3)=O)C2)cc2cc(C)cc(C)c2[nH]1 C(=O)(C1CSc2ccccc21)NC1COCCN(C(C2C(C(=O)OC)C2)=O)C1 C1(CNC(Cn2c(C)cc(=O)cc2)=O)CC2(CO1)CN(C(C1CC(C)(C)O1)=O)C2 CC1=C(C(=O)NCC23CCC(CN(C(=O)C(C4CCOCC4)C)C2)C3)SCCO1 C1(C)(C(=O)NCC(CC)NC(=O)CCCNC(=O)C(C)(C)C)CCCC1C C1(CCC)CN(C(C2CCS(=O)CC2)=O)CC1NC(=O)CC1CCCC1OC C#CC1(C(=O)NCC2CCN(C(C)=O)C2)CC(=O)C1.C1(CCC)C(=O)N1 C(=O)(CCCCCCC(=O)NCC1CCN(C(c2coc(Cl)n2)=O)CC1)OC C1(C(N2C(Cn3cc(CN(C(C)=O)C)nn3)C=CC2)=O)CC2(CC2)CO1 C1(C(N2CCC3C(C(=O)Nc4cc(CCC)ncc4)C32)=O)CC(=O)N(OC)C1 C1(C(N2CCC(N(C(CN(CCC)C)=O)C)C2)=O)CC(C)N(C)C1 N1(C(c2ncn(C(C)C)n2)=O)CCC2(CCC(N(C(=O)C=CBr)C)CC2)C1 C(=O)(C(CC)CCCC)N1CCN(C(C(C=CC)O)=O)CC1 c12cccc(c1)OCC(CO)NC(=O)C2(F)F.C(C(=O)NCCOC)OCCOC C12CC(C13CCC3)CN2.C(c1ccsc1)=C1CN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(CNC(C(C)SCCCC)=O)CCOC)cncc(Cl)c1 C1(CN(C(=O)C=COCC)CC)CCCN1C(=O)CCNC(c1ccoc1)=O N1(C(COCCCOC)=O)CCN(C(C2(Br)CC2(C)C)=O)CC1CCO C1(NC(C(c2cnn(C)c2)NC(C(CC)SC)=O)=O)CCCCCC1F Nc1cc(CN2CCCCC2CC(O)C(F)(F)F)ccc1Cl c1(C(c2nnnn2CC2CCOCC2)NCC2C(C)(C)C2)ncccc1F C(=O)(C(C)(C)C(N)=O)NC1CCCC(NC(C(C)c2ccco2)=O)C1 C1(NC(C(C(=O)OCC)C2CCC2)=O)CCN(C(=O)C=C(C)Cl)CC1C1CC1 c1(CC2CC(C)N(Cc3ccccc3)C2)ccccc1CNCC1=CCCCC1 c1(C(=O)OCC)[nH]cc(C)c1C(=O)N(CCNC(C1CC(C)(C)CO1)=O)C1CC1 C1(OC)CC(CSC)N(C(=O)C(C)Nc2ccc(N3CCCS3(=O)=O)cc2)C1 c1(C(=O)NC(CC)CNC(c2cccc(CC)c2F)=O)c[nH]c2cc(F)ccc12 Cc1cc(C(=O)NCc2cn(C3CN(C(=O)CCC(N)=O)C3)nn2)ccn1 N1(C(C2CCC(=O)O2)=O)CCC(NC(c2c(Cl)csc2Cl)=O)CC(O)C1 C(=O)(C1=CS(=O)CCC1)NCC(C)N(C)C(c1ccc(C(=O)C(F)(F)F)cc1)=O C1(C=C)(C(=O)NCC(CC=C)(C)CO)CCN(C(c2ncncc2N)=O)CC1 N1(C(CC2C(C)CCC2)=O)CC(C2CC2)(C(=O)NC2CCN(C(C)C)C2=O)C1 c1(OCC)cc(C(N2CCCC2)=O)c([N+](=O)[O-])cc1CNc1cnc(F)c(Cl)c1 C(C(O)C(=O)NCCC1CCCN1C(=O)C(C)CC1CCC1)OC N1(CCC)CCCC(C(=O)NCCCCCNC(=O)CCCn2ccnn2)C1 N1(C(CCC)=O)CCCCC1C(C1CCN(C(=O)C2=CCC2)CC1)CC(=O)NC O=C(C1=Cc2ccccc2C1O)NC1CN(C(=O)C2=C(Cl)CCCC2)CC1O c1(OC)cccc(S(=O)CC(=O)NCC(O)CCNC(c2coc(C)c2)=O)c1 c1(N2CCC3(N(C)CCC3)C2)[nH]c(=NCCCCS(C)(=O)=O)nc2scnc12 C(=O)(C1CCCc2nccn21)N(C)CC1N(C(c2c(C)cc(Cl)cc2)=O)CCC1 c1(OC)ncc(CN(C2CCCN(C(=O)Cn3nccn3)C2)C)cc1Br c1(C(=O)OC)nccc(NCC(C)NC(c2ccccc2C(=O)N(C)C)=O)n1 N1(C(C(C)SCC)=O)CCOCC1CC(N1CCC(COC)(OC)C1)=O Cc1cc(C)c([N+](=O)[O-])cc1C(N1CCC(C(N2CCC(O)C(C)C2)=O)C1)=O C1(C)(CNC(C(CC)=CCCC)=O)CCN(C(C2(OC)CCC23CCC3)=O)CC1 CC(CCC(=O)N1CC(CO)C1(C)C)NC(c1cccnc1)=O c1(C(=O)NCc2cn(CCC3(COC(C)OC)CC3)nn2)cc(C)nc(O)n1 N1(C(CONC(=O)C(F)C2CCC2)=O)CC2CCC=CC12 CC1(C2(C(N3CC(CC4CCCO4)C3)=O)CC2)CC1.c12ccc(o1)CCC2=O CCCCCCC(CC)NC(C1CCN(C(c2cn(C)cn2)=O)C12CCC2)=O C=CCC(C(=O)N(CC(C)N(C)C(c1cc(C(C)(F)F)n[nH]1)=O)C)C(C)C C1(C(=O)NC(C)C(CO)NC(c2ccc(C(F)F)s2)=O)CCC(F)(F)CC1 N1(C(C2CC3(CC3)CO2)=O)CCC2CC2(C(=O)NC2CC(O)CC2O)CC1 C(=O)(C(O)CC(N)=O)N1C(CNC(c2cccc(OC)n2)=O)CC(O)C1 C12(C(N(C3CN(C(=O)CC4OCCCC4(C)C)C3)CC)=O)C3C4C1C1C2C3C41C c1(SC2CCN(C)C2)ccc(C(=O)NCCC2CN(c3nncs3)CCO2)cc1 C(CCCCC(=O)N1CC2CC2(CNC(=O)CC2CCSCC2)C1)SC c1(C(N(CCNC(c2c(C#C)cn(C)n2)=O)C2CC2)=O)cc2[nH]nc(C)c2cn1 CCC(C)CCC(=O)NC(C1(C(=O)NCC(C)CN2CCCC2)CC1)C C1(NC(=O)Cn2ncnn2)(CO)CCCN(C(C2(c3ccccc3)CC2)=O)C1 c1(OC)cc(C2CCCN2C(=O)NC(C)(C)CC2CC2)ccc1O N1(C(CCC)=O)CCCCC(CNC(C2CCC(=O)N2C)=O)C1 c1(OC)c(C)cc(CNC(c2ccc(Cl)cc2OC)c2nnnn2C)cc1C CCC(CC)C(=O)N(C1CCCC1)CCNC(c1cnn(C2CC2(F)F)c1)=O C1(C(=O)NCc2ccc(O)c(F)c2)COC2(C1)CN(C(=O)CCC1CCCC1)C2 C12COCCN1C(=O)C(=O)NCc1ccc2o1.Cc1ccoc1C(F)(F)F c1(-c2cn(CC(CNC(c3nccc(Cl)c3F)=O)OC)nn2)cc(C)cc(C#N)c1 N1(CC2CC(=O)NC2)CCN(CC2CCCCO2)C(=O)C1 CC1CC(CNC(c2csc(Cl)c2)=O)CN(C(c2ccc(O)cc2)=O)C1 CC1CCN(C2CCN(C(=O)CC3CCCC3C(F)(F)F)CC2)CC1 C(=O)(C1=CC(C)(CC)C1)NC1CC(CNC(CCc2nnc(C(C)C)o2)=O)C1 CC(C)(C)CC(O)C(=O)N1CCC(CNC(c2cc(O)ccc2Cl)=O)C1 C1(F)(C(=O)NC(c2scc(C)n2)CO)CCN(C(=O)CC(C)CNC(N)=O)C1 C1(NC(c2ccc(CCC)s2)=O)CC(OC)CN(C(=O)CCCC(F)F)C1 CC1(C(N2CCOC(CNC(=O)CC3CCCC3)C2)=O)CCCCC1 N1(C(CC2C(C)C2)=O)CCC(CNC(=O)CS(=O)(=O)Nc2ccccc2)(OC)C1 N1(C(c2n[nH]c(C)c2C)=O)CCC(C)(C)C(C(=O)NC2COCC2F)C1 C1(NC(C2(C)CC(=C)C2)=O)CCN(C(=O)C(C)N2CC(C)C2)CC(O)C1 C1(CNC(C(CN(C)C)(F)F)=O)C(C2CC2)CCN1C(=O)C1=CCCCCC1 C1(COC)(CNC(=O)Cc2cc(Cl)n(C)n2)CCN(C(=O)C(F)(F)CO)C1 N1(CC(=O)NC(C)CNC(c2conc2C2CCCC2)=O)CC(=O)NC1=O C1(NC(C(C(C)=O)OCC)=O)CCCC(Nc2nc(COC)no2)C1 C1(C(=O)NC(C)CCO)Cc2ccccc2CN1C(c1ccc(O)c(Br)c1)=O c1(C(=O)NC23CC(NC(=O)CCSC(F)(F)F)(C2)C3)cnc2c[nH]nc2c1 c1(C(=O)NCCC(C)NC(C(CC)O)=O)cc(Cl)ccc1SC(C)C c1(SCC)ccc(C(N2CCC(N3CCN(C(=O)C=CBr)CC3)C2)=O)cc1 C#Cc1c[nH]nc1C(=O)NC12CC1CN(C(C1(c3ccccc3)CCC1)=O)C2 c1(NC2C(CCCC)CCC2)ncnc(NCCCc2cnn(C)c2C)c1C c1(C(=O)NCC2(c3ccc(Cl)cc3)CC(O)C2)cc(Cl)c(O)c(Br)c1 Cc1cc[nH]c1C(=O)NC(Cn1ccnn1)C(=O)N1CC(C(N)=O)(CO)C1 Cc1cnc2cc(C(=O)NC(C)C(CO)NC(c3cc4ccsc4s3)=O)ccn12 CC(c1ccco1)=CC(=O)NCCOC1CN(C(c2cc(C(C)C)sn2)=O)C1 N1(C(CC(C)C(F)F)=O)CCCC2(CCN(C(=O)C=C(C3CC3)C3CC3)C2)C1 C#CC1(C)CCN(C(=O)C(C(C)C)NC(=O)CCC2CCCO2)CC1 C1(NC(c2c(C)ccc(C(=O)OCC)c2)=O)CN(C(=O)CCSC)C2(CCC2)C1 N#Cc1cccnc1-c1cn(CCCCC(N2CCC(C3CCCO3)C2)=O)nn1 C(C(C)NC(=O)Cc1cc(C)cs1)(C(C)C)NC(COCCC)=O Nc1[nH]c(=O)c(Cl)nc1C(=O)OCc1csc(-c2ccco2)n1 C1(CC(=O)NC2CCN(C(=O)Cn3cncn3)C2C)(C(=O)OC)CCCCC1 C(=O)(C#CC1CCOC1)NCC1=NOCC1.CN1CCC2(C1)C(=O)N2 CC(C)CC(F)C(=O)NCCC1(NC(=O)C(C)Sc2ccccn2)CC1 Cc1nn(C(F)F)cc1S(=O)(=O)N1CCC2C(C1)CN2c1nnnn1C(C)C N1(C(=O)COc2ccccc2Cl)CC2CCC1CN2C(=O)C1=CCCS1 c1(C(N2CCC(NC(c3occ(C)c3)=O)CC2)=O)cccc([N+](=O)[O-])c1Cl C1(NC(CCC=C(C)C)=O)CN(C(c2sccc2CN(C)C)=O)CC2CC12 N(C(=NCCCOc1ccccc1)NCc1ccccn1)Cc1n(C)ncc1Cl C1(C(=O)NCC2CCCN(C(C3CC4C=CC3C4)=O)CC2)CCc2nnnn2C1 C1(NC(COC(C)=O)=O)CC(CNC(C2CC2c2cccnc2)=O)CC1O c1(OC)cccc2c1OC(C(N1CCN(C(=O)CC3OCCO3)CC1CF)=O)C2 c1(C(=O)NCCN(C(C(C2CCC(=O)N2C)C)=O)C2CC2)cnc2n1CCC2 C1(NC(C=Cc2ccc(C)s2)=O)CC2CCC1N(C(C1C(C)C1(F)F)=O)C2 C(CC1CCC1)(C(=O)N(C1(C(=O)NCCc2cc(C)on2)CC1)C)OCC N12CCCC(C1)c1ccc(cc1)NC2=O.n12nccc1C2.C(C(C)C)OCC C(=O)(CCCSCC)N(C(=O)C(C)n1cccc1)C(C)C.Cc1cscn1 C12(C(=O)NC3C(C)CSC3)CC(CN1C(=O)CN1CCCC1)C2 C(=O)(CC(C)(C)C(=O)NCC1CCC(NC(=O)Cc2sc(S)nc2C)C1)OC CC1(C)CCC(CNC(c2c[nH]nc2CNC(c2cc(O)nc(O)n2)=O)=O)CC1 C1(NC(C2Cc3nncn3C2)=O)CC12CCN(C(C1CCN1)=O)CC2 C12(CCNC(CNC(=O)NC)=O)CCC1CN(C(=O)C(C)(C)C(F)F)C2 N1(C(C(COCC)N=[N+]=[N-])=O)CCCC2CN(C(c3cccc(=O)n3C)=O)CC12 Cn1nc(C(=O)NC2CCCC(NC(=O)CN3C(=O)CCC3=O)C2)cc1C1CC1 C1(CNC(C2CC2(F)F)=O)CC2(CCOCC2)CN1c1ncnc2c1SCCC2 c1(C(N2CCCC(n3cc(CCC(N)=O)nn3)C2)=O)cc2cc(Br)sc2s1 c1(C(N2C3CC(NC(C=C(C)c4cccs4)=O)C3CC2)=O)cnc2c(c1)CCC2 CC(C)CCCCCC(=O)N(C1CN(C(=O)Cc2cc[nH]n2)CC12CC2)C n1(CC)ccnc1CCC(=O)NC1(C)CC(C(=O)N)C1.c1(C2CC2C)ccn(C)n1 c1(OC)nccc(C(=O)NCC2(O)CCN(C(C3CC(C)C3)=O)C2)n1 c1(NCC)ccc(C(=O)NCCOCCCN(C)C(C2CCN(C)C2C)=O)cn1 N1(C(c2c(C)noc2)=O)CCC2(C1)CN(C(C1CC3CCCCC13)=O)CCO2 Cn1nccc1C=CC(=O)NCc1nocc1C(N1CCC1(C)CCO)=O N1(CC)CCOCC1C(=O)NCC1(C(=O)N(C)OCC(F)(F)F)CC2(CC2)C1 C1(C(=O)NCCC2N(C(c3c(C(C)C)noc3)=O)CCOC2)CC2CCC(C1)S2 c1(C(=O)NC2(C)CCN(C(c3ccc(C(C)=O)o3)=O)C2)cccc(C2CC2)c1Cl C(=O)(CC(CNC(C1CCC1(F)F)=O)C1CCC1)NC(CCCN(C)CC)C C#CC1(C(=O)NC(C)CCC2CC2)CN(C(=O)C(CC)CC)C1 C1(OC)CN(C(C2CC3CC3C2)=O)CC1NC(=O)C(C1(O)CCCC1)F N1(C(=O)Nc2c(C(=O)OC)cc(F)cc2)CC2CC3(CCC3)C2C1 N1(C(c2ccc(C(C)C)o2)=O)CCC(CO)(NC(=O)C=Cc2cn(C)cn2)C1 c1(C(=O)NC(C2CCCC2)C#C)coc(CNC(C2(Cl)CC2)=O)n1 C1(CNC(C(C)CC(N)=O)=O)CC2(CO1)CN(C(C1CC(OC(F)(F)F)C1)=O)C2 S(=O)(=O)(c1c[nH]c2nc(Cl)ccc12)N1CCC(C)(CC(C)C)CC1 C1(C(N(C)CC2CCC(=O)N2)=O)CN(C(=O)Cc2ccns2)CC12CCC2 C1(CCNC(=O)CN2CC3CC3C2)(OC)CN(C(=O)CCCC2CC2C)C1 c1(C(=O)NCC2CCN2C(=O)Cn2cnc([N+](=O)[O-])c2)cc2cccc(F)c2o1 Cc1ccoc1CC(=O)NCC1CCC1NC(c1csc(-c2ccccc2)c1)=O C1(NC(c2n[nH]c(CC)c2Cl)=O)CCC2CCN(C(=O)CC3CC3)C1C2 c1(SCC)ccccc1C(=O)NCC12CC(CNC(C3CCC3C)=O)(CO1)C2 c1(N(CCN(C(C(C2CCOC2)OC)=O)C(C)C)C)snc(Cl)c1C#N c1(C(=O)NC2CCN(C(c3ccccn3)=O)C2)ccn2cnnc2c1 C1(OC)CCN(C(=O)CC2(O)CCN(C(=O)Cn3ccnn3)CC2)C1(C)C Cc1cnn(CCC(=O)NCC2CCN(C(=O)CSC3CCCCO3)C2)c1 N1(S(C(C)C)(=O)=O)CCC2(CC1)CC2C(N1CCC(N(C)C(C)=O)C(O)C1)=O CC(C(C)(C)CN(C)C)NC(=O)CNC(=O)CNC(=O)CC1OCCCO1 C(C(C(=O)Nc1ccc(C)n(C)c1=O)C(C)(C)C)NC(c1cc(CC)on1)=O N1(CC#C)CCC(Nc2ccc(COC(=O)CC)c(C)c2)C(C)C1 N1(C(c2c(C#N)scc2)=O)CCC2(CCCCC2NC(=O)CNC=O)C1 C(=O)(CC(C(F)(F)F)OC)NCCN(C(C(C(CC)O)C)=O)Cc1ccccc1 N1(C(C(C)CC2CC2)=O)CC2CC(C1)C2NC(c1ncsc1-c1ccccn1)=O C1(CNC(C2(CC=C)CCN(C(C3CC3(C)C(F)F)=O)C2)=O)OCCCC1(C)C Cc1ccc(C#N)c(N2CCCC(CNC(=O)Cc3nc(C4CC4)nn3C)C2)n1 c1(C(C(=O)NC2COC2)N(C2CCC2)Cc2n(C)cnc2)cccc(Cl)c1 N12CCCN(CC1)C(=O)c1ccccc1C2.c1(C(=O)OC)ccc(OC)s1 O(N(C)C(=O)C(F)CC1CN(C(=O)CC2CCCCCC2)C1)CC(=O)OC N1(C(c2c(CC)nco2)=O)CCC(N=c2[nH]c3ncc(Cl)cc3o2)C(C)C1 C1(C)(C(=O)NC23CN(C(C(CC)OC)=O)C(CC2)C3)CC(C2CC2)=NO1 N1(C(CS(=O)(=O)NC)=O)CC2(CNC(C3C4CCCC34)=O)CC1CO2 c1(N2CCC(NC(c3ccc(C)c(C)c3)=O)C(C)C2)ncnc2c(C)csc12 S(=O)(=O)(c1ccc2c(c1)NCC2)N1CC(c2cc(C)no2)C1 C12(C(=O)NCc3c(OC)cc(C)s3)CC(C)(CN1C(=O)C(C)CC1CC1)C2 c1(N2CCC(=C)C2)nc(N(CC(C)C)C)c2c(n1)CSC2.N(C)C(C1CC1)C1CC1 Cc1c(C(N2CC(C(=O)NC(C)(CO)C3CCCC3)C(C)C2)=O)ccn1C CC(C)C(C)(C)C(=O)NCc1ocnc1C(=O)NC1CN(C)CC1(C)C C(=O)(C1CCc2sc(NC(=O)C(C)(C)CC3CC3)nc21)C(=O)OCC.C1CO1 N1(C(CCc2cnc(C)o2)=O)CCCC(C)C1CNC(c1cncnc1)=O CCC(CC)CC(=O)N1CCN(C)C(CNC(=O)C(C(F)(F)F)OC)C1 c1(CCC(N2CCC(NC(c3cccnc3F)=O)C2)=O)cccc(Cl)c1Cl CC1(C)CNC(=O)OC12CN(C(c1cc([N+](=O)[O-])cnc1O)=O)C2 C1(C(=O)NC2CCC(C)N(C(=O)C3=C(Cl)CCCC3)C2)CCC2(CCOCC2)C1 C=C(Cl)C(C)(C)C(=O)NC1COCCN(C(c2cnc(C(C)O)s2)=O)C1 C1(C(=O)NCCCN(C(C2(CC)CCCO2)=O)C2CC2)CN(C)C(=O)N1 N1(C(c2cc(-c3ccco3)c[nH]2)=O)CC(CNC(C23CCCC2C3)=O)C(O)C1 c1(SCC(=O)NC2(CNC(Cn3ccc(C)n3)=O)CCC2)nc2ccccc2o1 N1(C(C(CC)=CC)=O)CC2CCCC(NC(C3CCCCC3C)=O)C2C1 C1(C)(COC)CN(C(=O)C(C)(c2cccs2)NC(=O)CC(C2CCSC2)SC)C1 C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCCC(O)(CNC(Cc2cnc(C)[nH]2)=O)C1 C1(C(=O)NCC2C(NC(c3ccc(CC)[nH]3)=O)CCC2)CCC(=O)N(C)C1 C1(=O)NNC(=O)CCN1CC(F)(F)F.N#CCCS(=O)(=O)N N1(C(c2c(C)[nH]cc2)=O)CCC(N(C(=O)C(C)OCC2CCCO2)C)CC1 Cc1c(C(N2CCC3CCN(C(=O)Cc4cccs4)CC23)=O)sc2ccccc12 C1(C(N2CCCC(CNC(CC(CC)O)=O)C2)=O)CCc2nncn2CC1 C(C(C)(F)C(C)C)NC(CN(C(=O)C(CCOC)OC)CCC)=O C(=O)(C1CCc2c[nH]nc21)NCc1occ(C(=O)NCCCCNC(N)=O)c1 CCC(C(C)CN(C)C)NC(=O)C(CC1CCC1)NC(c1cncc(NC)c1)=O C(c1cncc(F)c1)=CC(=O)NC1CC(CNC(C2CC(OC)C2)=O)CC1O C1(CC(C)NC2CCN(Cc3nnc(-c4ccccc4)o3)C2)CCC(C)CC1 C1(CNC(c2cc(N)c(F)cc2)=O)CC12CCN(C(C1CCCN1N=O)=O)CC2 c1(C(N2CC(OCCNC(CC3C(C)(C)CCC3)=O)C2)=O)cc(N)cc(F)c1 Cc1cc(CNC(=O)COCCNC(c2[nH]nnc2C)=O)cc(O)c1 Cc1cccc(C)c1OCC(O)CN1CC2CC1CN2NC(=O)CC(C)C1CC1 C1(C(=O)NC2C(C)CCN(C(C3(O)CCSCC3)=O)C2)CCC2C(CC1)C2(F)F N1(C(c2c(CC)scc2)=O)CC(NC(=O)CNS(=O)(=O)C2CC2)C(C2CC2)C1 c1(C(N2CC(NC(c3ccc(O)nn3)=O)CC(C)C2)=O)c(Cl)cc(Cl)cc1Cl C1(CNC(C(C=CC)O)=O)CCCN(C(=O)Cc2csc3nccn23)CC1 c1(C(N(C2CN(C(=O)C=CBr)C2)C)=O)csc2cccc(F)c12 C=CC(F)(F)C(=O)N1CC2CC1C2C(=O)NC(CCO)C1CC1 N1(C(c2c(C)nc(CCC)s2)=O)CCN(C(=O)CCN2CCCC2)CC1C1CC1 c1(C(=O)NC2(CCNC(C(CC)N(C)C)=O)CCOCC2)cccc2ncnn12 C1(C)(NC(CN(C(=O)Cc2ccns2)CC#C)=O)CCC2(CC1)CC2 c1(C(=O)NCCNC(CCOCC#C)=O)cc(Cl)c2c(c1)OCCCO2 C1(O)(CCNC(C(C(=O)OCC)OC)=O)CCN(C(c2ccc(Cl)[nH]2)=O)CC1 CCC(C)(COC)CC.C1(=O)C(CCNCCN(C)C)O1 N1(C(c2ccc(OC)o2)=O)CC2(CCCC2NC(c2ccc(CC#N)cc2)=O)C1 C12(NC(c3ccn(C)n3)=O)CC3CCC(C1C2)N3C(c1cnc(N)c(CO)c1)=O N#CC1CCCCC1NC(=O)C(CNC(c1cc(C(N)=O)co1)=O)NC=O C1(NC(CC2C(C)=NN(C)C2=O)=O)COC2CN(C(=O)Cc3cnco3)CC12 CC1CN(C(c2ccoc2CNC(C2COC(=O)N2C)=O)=O)CCO1 C1(C)(CNC(COCCC)=O)CCCN1C(c1cn(C)nc1SC)=O CCC(C)(O)C(=O)N1CCC(Cn2cc(-c3ccccc3OC)nn2)C1 C(=O)(C(O)C(F)(F)F)N1CCCC(CC(=O)NC(C23CCC(CC2)C3)C)C1 C1(CNC(C2CCN(C(c3ccccc3NC)=O)C23CC3)=O)CC2CCCC2C1 C1(NC(COCC#C)=O)CCCC1(C)CNC(C1CCCN1C(=O)NC)=O N1(CC)C(C)CN(C(=O)CCNC(C2CCCCC(=O)C2)=O)CC1C N1(C(CC=C(C)C)=O)CC(NC(=O)Cc2ccc(CC(C)C)cc2)C2CC2C1 c1(C(N2C(CNC(C3C=CC=CC=C3)=O)CC(O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] CCC(C)CC(C(=O)NOCCC(C)O)NC(=O)C=Cc1ccco1 n1(CC(=O)NC(C)C(CO)NC(=O)CC(F)(F)C(F)F)cnc2sccc2c1=O C1(CNC(CN(CC(F)F)C)=O)OCCC1C(=O)NC1(n2ccnn2)CC1 c1(C2C(CN3C(CN(C)C)CCC3)C2)ccc(F)c(F)c1.C12CCCN1C2=O C1(NC(C=CC2(C)CCOCC2)=O)CCC2(CCN(C(C3CCOC3)=O)CC2)C1 Cc1c(C(=O)N(C2CN(C(=O)Cn3cccc3)CC2(C)C)C)ccc(F)c1F CC1C2CCC(C2)C1C(=O)NCCn1ccc(C(N2CC(C3(C)CC3)C2)=O)c1 C12(NC(c3nc(C)sc3)=O)CCCC1N(C(C1(C(F)(F)F)CC=CC1)=O)CC2 N1(C(C2(c3c(C)cccc3)CC2)=O)CC2CC(NC(c3csc(C)c3N)=O)C(C2)C1 CCC(O)C(=O)NC(CNC(=O)CCNC(=O)OC(C)(C)C)C1CC1 C(C(C(=O)NCCCN(C1CCCC1)C(=O)C=CC=C(Cl)Cl)OC)OC c1(OCC(=O)N(CCC(C)NC(c2ccc(CC)o2)=O)C)c(C)occc1=O C1(NC(C2C(C=C)OCC2)=O)CC1C1CCN(C(c2ccnc(C)c2N)=O)CC1 C(CCC(C)C(=O)NCC(F)F)OC.c12cccc(c1)OCC(=O)N(C)C2 C1(NC(C2(COCC)CC2)=O)CN(C(=O)C=Cc2cn(C)cn2)CC1C(F)F N1(C(C2CCC(=O)N2)=O)CC2CCN(C(c3ccncc3Cl)=O)CC(C2)C1 c1(CC)cc(C(=O)OC(C)C(c2ccccc2OC)C)cc(CC)c1 c1(ONC(c2c(F)ccc(Cc3n(C)nnc3)c2)=O)cncc(S(C)(=O)=O)c1 c1(C(N(CCC(C)NC(C(CC)C2CCOCC2)=O)C)=O)ccccc1Cl NS(=O)(=O)c1c(C(=O)NC2CC(NC(=O)C=CCO)C2)ncc2ccccc12 Cc1nn(C)c(=O)c(C(=O)NC2CC2CNC(=O)CC2C=CS(=O)(=O)C2)c1C Cc1cccc2nc(C(=O)NC3(CO)CCCN(C(=O)CCCC4CC4)C3)cn12 C1(C(N2CC3C(CNC(CN(c4ccc(Cl)cn4)C)=O)C3C2)=O)COC2(CCC2)C1 C(=O)(CCS(C)=O)N(CCCNC(Cc1ncc(C)[nH]1)=O)Cc1cccnc1 CN1CC(C)(C(N2CCCOC(CNC(c3cc(Cl)ccc3F)=O)C2)=O)CC1=O c1(OC)ccc(C(C)C(=O)NCC(=O)Nc2cccc(Cl)c2)cc1 C(=O)(C(C(C)(C)C)N(C)C)NCC1CCC(C(NOC(COC)COC)=O)C1 c1(CNCC(C2CCOCC2)OC)cc(Cl)cc(F)c1O C1(C(=O)Nc2ccc(F)cc2)(CN2CC3N(C(C4(Br)CC4)=O)C3C2)CCOCC1 N1(C(c2cnc(=N)[nH]c2)=O)CCC(C2CCN(C(=O)Cc3ccns3)CC2)C1 c1(C(c2n(CC#C)nnn2)NC(c2cncc(F)c2)C)c(F)cc(C#C)cc1F N1(C(CCC)=O)CCCCC(CNC(C2CC2C2CCC2)=O)C1 N1(C(C=CCCC=C(C)C)=O)CCCCC1CCN(C)C(C1(C)CS(=O)(=O)C1)=O C1(C(NOC(C)C)=O)CC2(C1)CN(C(c1cc(F)c[nH]1)=O)C2 C1(CNC(C2C(C)C2)=O)CCC2(CC1)CCN(C(=O)COC(F)(F)F)CC2 C1(NC(C2(C(C)C)CCC2)=O)CC2CCCC(C1)N2C(C1COC(C)(C)C1)=O C1(C2CCN(C(C3CCCCC34CC4)=O)C2)(NC(c2ccn(C)c(=O)c2)=O)CC1 C1(C(C)C)C(=O)N1.c1(C(=O)NCCNCC)ccccc1OC(F)(F)F Cc1c(C(=O)N(CC(O)CNC(C2CC2c2cccs2)=O)C)ccn1C1CC1 N1(C(C(n2ccc(C)n2)C)=O)CCN(C(=O)C(C)(C)N=[N+]=[N-])C(C)C1 C(CN=c1ccc(S(=O)(=O)N2CCC(CCC)(CO)C2)c[nH]1)N(C(CC)C)C CC1(C(N2CCC(NC(c3ccc(C#N)o3)=O)CC2)=O)CCOCC1 c1(C(=O)NCC2C(CC(=O)NC(C#C)C)C2)cnn(C)c1C c1(CNC(C(C(C)OC)O)=O)cc2n(n1)CCN(C(C13CCC(CC1)C3)=O)C2 Cn1cnc2cc(C(N3CCC(CNC(=O)COC4CC(F)(F)C4)C3)=O)cnc12 C1(NC(c2c(C(=O)OC)nn(C)c2)=O)(CO)CCCN(C(=O)CS(N)(=O)=O)C1 C1(NC(CCOC)=O)CN(C(=O)C(F)CC2CCCCC2)CCC12CCC2 c1(NC)cc(Cl)ccc1C(=O)N(CCCN(C(=O)COCC1CCCO1)C)C C=CCCCC(C(=O)N(C)C)N1CCC(OCC(=O)OC)C1 C(=O)(C(C(=O)N(CC(C)NC(C1CCN(CCF)CC1)=O)C)C1CC1)OCC CN(CP(C)(C)=O)CC(C1CC(C)(C)C1)O N1(C(C(CC)(C)C)=O)CCCN(CCNC(=O)C(COC)CC)CC1 C1(NC(c2n(CC)nc(C)c2)=O)CCOC12CCN(C(=O)C(C)(O)COC)CC2 CCC(C)C(O)C(C)C(=O)NCCCC1(NC(C2CC2C(N)=O)=O)CC1 C1(NC(=O)Cc2ccon2)CN(C(C2(c3ccno3)CCOCC2)=O)CC12CC2 C(C)(C)(CCC(=O)N1CC(C)(CCC(=O)NC2CC(C)CCC2O)C1)OC N1(C=O)CCC2(CC1)CCN(C(=O)CN1CCCCC1)C2.C1(=O)CCN1C(C)C.CN C(N=c1[nH]c(=NCC(C)(C)C2CC2)c2cccc(F)c2[nH]1)c1c(C)nc(Br)s1 Clc1ccccc1-c1noc(-c2cccn2CC2=NC(Br)=C(I)C2)n1 C(CCC(C)C(=O)N1CCCC1CNC(c1cccnc1OCCO)=O)OCC N1(C(c2c3ncn(C)c3ccn2)=O)C2CCCC1CC(O)C2 c1(C(=O)NCCn2c(CC)ncc2)oc(CNC(=O)C(C)(Cl)Cl)nc1C c1(NC(CC)CCOC)ccc(S(=O)(=O)NCCC2CC3CC3C2)cc1Cl N1(C(CC2(CNC(C3CC3(F)F)=O)CC2)=O)CCc2cc(F)ccc2C1 c1(C(=O)NCCN(C(C2CC(C(C)C)C2)=O)C(C)C)ccncc1 N1(C(C(C)(C)N(C)C)=O)CC(CC(=O)NCC2CCCC(CO)C2)C2(CC2)C1 CC1CC(NC(=O)C(C2(O)CN(C(c3ncccc3O)=O)C2)F)CCN1C C(S(=O)CC(=O)Nc1ccc(OC2CCC2)cc1)c1onc(CC=C)n1 n1(C(C)C)cnc(C(=O)NCC2CCC2NC(c2ccsc2-n2cnnn2)=O)c1 C(=O)(C1=CC2(CCOCC2)C1)N1C(C)(CC)CC(NC(=O)CNC(=O)C2CC2)C1 N1(C(c2cc3cccc(C)c3o2)C(=O)NCCCC)CC=CCC12CCCCC2 C1CC(N(C)C)C(=O)Nc2nnsc2C(=O)N1.C(=O)(CCOC1CC1)NCC C1(C(=O)NC2CCN(C(c3cc(C(C)(C)C)ncc3)=O)C2)CC2(CCCC2)C1 c1(C(=O)NC23CC(C2)N(C(C2CCC(F)(F)C2)=O)C3)ccc2nonc2c1 CCCCC(O)CC(=O)NC(CCC1CC1)C(=O)NCc1cncc(F)c1 c1(-c2n(CC)nc(Cn3cc(C)cn3)n2)ccc(S(=O)(=O)N2CCCC2)cc1 c1(-c2cccc(C)n2)ccc2c(C(N3CCCC4CC34)=O)cnn2c1 c1(C(=O)NC2(C)CN(C(c3n(CC)cc(Cl)c3)=O)C2)ccc(F)c(F)c1N C1(N(C(CN(CC)CC)=O)CCO)CCCN(C(=O)Cn2nccc2C)C1 N1(C(CC)=O)CCCC2(NC(=O)C=C3CCCC3)CC2C1 C(C(C)CC(=O)NCc1nnn(C)c1C)NC(c1n(CC)nnc1)=O N1(N(CC)Cc2ccccc2Cl)CCC(C)(NC(C2CC(O)C2)=O)CC1 C(=O)(C(C)(C)C(C)C)N(CCC(=O)N(CCOCC(=O)NC)C)C C(CC(=O)N(C)CCN1CCOC1=O)(C(C)OC)NC(C1(CCCC)CC1)=O CC1CCN(C(=O)C=Cc2cscn2)CC1NC(c1coc(C(F)F)n1)=O c1(C(N2CC3(C(CNC(C(CC)(C)O)=O)C3)C2)=O)ccc(N2CCCC2)c(F)c1 C(=O)(C(C)(O)C(F)(F)F)N1CCC(=C(C)C(=O)N2CC(SC(F)(F)F)C2)C1 Cc1nc(C(=O)NCc2cc(C(=O)N(C)C)no2)cn1C.C12CC1S2 c1(C(N(C(=O)COC(=O)CCC2CC2)CC)C)ccc(C(N)=O)cc1 N1(c2nnc(C(C)(C)C)o2)CC(NC(C2CC(C3CC3)=NO2)=O)C2CCCCC12 c1(C(=O)NCC(CN(C(=O)CCCNC(=O)C(C)(C)C)C)O)cnn(C)c1 N1(C(CCc2n(C)ncc2)=O)CCC(C(N2CCC(CN=[N+]=[N-])C2)=O)(CO)C1 c1(C(=O)Nc2ccc(OC(c3ccc(Cl)cc3)C)nc2)cnc(C(C)(C)C)nc1 C1(NC2CC(CCS(C)(=O)=O)C2)CCCN(c2ccccc2F)C1=O C(=O)(C1=NNC(=O)C1)N1C(C2CCN(C(c3c(C)occ3)=O)CC2)CCC1 CCS(=O)(=O)c1ncccc1CNC(=O)NC(c1ccc(C(F)(F)F)c(Cl)c1)C N1(c2nc(C)c3n2CCC3)CCCC1C1CCCCN1C(c1ccnn1C)=O c1(C(=O)NC2CC(NC(C(C)NS(C)(=O)=O)=O)C(O)C2)cc(O)cc(C#N)c1 c1(OC)ccc2nc(C(N3CC(NC(=O)C(C)(C)SC)CC3(C)C)=O)ccc2c1 CC(F)(F)C(F)(F)CC(=O)N1CCC(CNC(=O)CSc2ccc(F)c(F)c2)C1 c1(C(=O)NCCCN(C(C2C(C)(CC)C2)=O)C)cc(C)nn1-c1ccccc1 C1(C(=O)NCc2cnc(C)s2)COCCN(C(c2coc(N(C)C)n2)=O)C1 N#CC1(C(N2CC3(C2)CN(C(=O)C=CC2CCC2)C3)=O)CC2CCC1C2 c1(C(=O)NC(CO)CO)cc(-c2ccc(F)nc2)c2n[nH]cc2c1 C(CC(O)C(=O)NN1CCCC1C(=O)NC1CCN(C(=O)C2CC2)CC1)SC C1(O)(C(C(=O)N(C)CC2(NC(CC3CC(CC)C3)=O)CC2)F)CCCC1 c1(C(=O)NC(C2CCN(C(C3N(C)CC(F)C3)=O)C2)(C)C)cnc2ccoc2c1 c1(C(N2CCC(C(=O)NC3C(C(C)(C)C)CC3)CC2)=O)cc(F)c(O)c(Cl)c1 C1(NC(CC2C(NC(C(C)N3CCCC3)=O)CCC2)=O)CC2(CCC2)C1O c1(C(=O)NCC=CCNC(=O)C(F)(F)c2csc(Cl)c2)ccncc1Cl C1(C2(NC(C3C(CN(C)C)C3)=O)CC2)CCCN1C(=O)CCC1OCCO1 C1(C(=O)NCC2(O)CCN(C(CC3C(CC)C3)=O)C2)CCc2nc[nH]c2C1 c1(OC)cc(F)c(Br)cc1C(=O)N(CCNC(c1cn(C)nc1C)=O)C1CC1 N1(C(c2cc(S(C)(=O)=O)sc2)=O)C2CCC1CN(C(=O)CC1CNC(=O)C1)CC2 C1(NC(=O)COCC2CC2)CCC(CCNC(c2cn(C3CCC3O)nn2)=O)C1 C1(CNC(C2=CC(C)C2)=O)CCCCN(C(C2CCCCO2)=O)C1 c1(CCC(N2C(CNC(c3ccc([N+](=O)[O-])o3)=O)CCC2)=O)c(F)cccc1Br c1(C(N2CCC(C(C)C)(C(=O)NC(C)Cn3cncn3)C2)=O)cnccc1C#N C1(C(=O)NCC(CC)(CC)NC(c2[nH]cc3c2CCC3)=O)CN(C)CC(C)O1 C1(CNC(c2c(C)cc(CO)o2)=O)CN(C(=O)CC2=NNC(=O)C2)C2CCN1C2 C1(SC)CN(c2ccnc(Cn3ccnc3)n2)CC1NC(C)(C)C N1(C(C(CO)NC(CCC(=O)NCC)=O)=O)CC2(CCC(=O)N2)C1 N1(C(CN(S(C)(=O)=O)C)=O)CCCC1C1CCCN1C(c1n[nH]c2c1COC2)=O C12(C(N3CCCC(CC(=O)N(C)CC4(N(C)C)CC4)C3)=O)CCC(C)(C1)OC2 c1(C(=O)NCC2(NC(C(CC(=C)C)NC(C)=O)=O)CC2)oc2ccc(Cl)cc2c1C c1(C(N2CCOCC(CNC(C=COCC)=O)C2)=O)cc(F)c(F)c(C#N)c1F c1(CNC(=O)Nc2n(CC)nc(C)c2)c(F)cncc1Cl C1(O)(CCNC(C(F)OC)=O)CCN(C(c2cnn(CCO)c2C)=O)C1 c1(Cc2cn(C3(NC(c4c(C)n(C)nn4)=O)CC3)nn2)cn2c(n1)CC(C)CC2 N1(C(COCCOC)=O)CCC(C)C1c1cn(CC2CCOC2C2CC2)nn1 CCCCCC(C)CC(=O)NC1CN(C(=O)Cc2c[nH]nc2C)CCC1O c1(C(=O)NCCCC(C(=O)N2CCC(C)(C)C2)O)ccc2n[nH]cc2c1 Cc1nc(O)c(C(=O)NCC2(O)CN(C(C3CC34CC4(F)F)=O)C2)nc1C C1(C(C)C)C(NC(c2cccc(Cl)c2)=O)CCN1C(=O)C(c1cccc(Cl)c1)C c1(C(=O)NC2CCCCN(C(C3(CCC)CCC3)=O)C2)ccc2c(c1)C=CCC2 c1(COC)ccccc1C(=O)NC1CC(C)N(C(=O)CCCn2ccnc2)C1 c1(C(=O)NC(CNC(C(CCC)OC)=O)C)cc(F)cc2nc[nH]c12 C1(NC(Cc2cccc(SCC)c2)=O)CC2CCC1(NC(=O)C=CC1CCC1)C2 Cc1c(C(=O)NC2CC(O)CN(C(=O)CCC3CCC3)C2)sc2ccc(F)cc12 c1(N(CC(=O)NCC(C)(C)C)C)cc(C(F)(F)F)cnc1N.N12CCN(CC1)CC2=O CC(C)C(F)(CNC(=O)CC1CCCN1C)C(=O)NC1CCCN2CCC1C2 Cc1nc2c(cnn2C(C)C)cc1C(=O)NC(C)(C)CCNC(=O)C(O)C1CC1 CC1C(CNC(=O)CCCN(C(=O)COCCCF)C)C1(F)F C12(C(N(CCCNC(C(N3CCC(C)CC3)=O)=O)C)=O)CCC(C#N)(CC1)CC2 C(=O)(C(C#N)CC)NCCC1(CNC(C(C=C)O)=O)CC1 Cc1ccc(Cl)cc1-n1cc(C2CCC2C(N2CC(CN3CCCCC3)C2)=O)nn1 Cn1ccc(C(N2CC(O)(C(F)C(=O)NCC3CCN(CCF)C3)C2)=O)c1 C(=O)(C(CO)C(C)(C)C)N(CCN(C)C(c1cn(C)nc1C(F)F)=O)C c1(OC)cc([N+](=O)[O-])c(Cl)cc1C(=O)NCCOCCNC(=O)C=CCC1CC1 N1(C(C(CC)(C)O)=O)C2CCC1CC(NC(c1cccc(=O)n1O)=O)C2 Cc1cc(F)c(Br)cc1C(=O)NCC1CCC(C)CN1C(=O)CC(F)F c1(N(C(CCOCCCNC(C2C(CCC)C2)=O)=O)C)cc(C)cc(C)c1 Cc1ccc(C(=O)NOCC(=O)NCC2(CO)CC23CCC3)cn1.C(C)C C(CN=C(NC1CC1C(C)C)N(C1CC(C)CC=CS1)CC1CCCCS1)OC c1(C(=O)NC23CC(NC(c4c(C)cc(CC)o4)=O)(C2)C3)c(C)nc2ccccn12 c1(C(=O)NC2(COC)CCN(C(C(C(=O)OC)OC)=O)C2)cnc2n1CCOC2 c1(C(N2CC(C)CC(NC(COC)=O)C2)=O)cc2c(Br)coc2cn1 CN1CCC(=CC(=O)NC2CC2NC(C2(CC(C)=O)CCCC2)=O)CC1 c1(OC)cc(O)c(CN2CC(C)(C(=O)NC(C)CN(C)C)C2)cc1Br C(C)(c1ccccc1)=CC(N1CCC(OCCNC(C2C(CCC)C2)=O)C1)=O C1(CC(=O)N(CCC(C)O)C)CCCN(C(=O)CN(C)C(=O)C2CC2)CC1 c1(NC(C2(C(=O)NCC3(CN(C)C)CC3)CC2)=O)ccc(C(F)(F)F)cn1 N1(C(c2ccc(C#C)o2)=O)CC2CC(C1)CN(C(c1coc3c1CCCC3)=O)C2 N1(C(CCC)=O)CCCC1C(=O)N(C(C)CN(C)C(c1cscc1Cl)=O)C N1(C(C2COC(=O)O2)=O)CCOCC(NC(C2(C(=O)NC3CC3)CC2)=O)C1 N1(C(c2cc(C)oc2C)=O)C2CCC1CN(C(=O)C1=CCCCO1)CC2 C1(C(=O)NCC#CC(=O)NCCC2(O)CCOC2)(CC)CCCC1 C(C(COC)C(=O)NCCCCC1CN(C(C2CC2c2ccccc2)=O)C1)OC C1(CNC(c2c(CC)c[nH]n2)=O)CCCCN1C(=O)CNc1ccc(O)cc1 CC(N=c1ccc(C2CCOCC2)n[nH]1)C(=O)NC1CC1c1ccc(Cl)cc1 C1(NC(CCc2n(C)ccc2)=O)CN(C(C2CCCN2C=O)=O)CC1(C)C N1(C(c2cn(C)nc2)=O)CCC(N=c2cc[nH]c(C#N)n2)C2(CCC2)C1 c1(SCCC(N2CC(NC(C(c3ccccc3)SC)=O)C2)=O)ccccn1 c1(N2CCCN(C(C)=O)CC2)ccncc1S(=O)(=O)NCc1cc(OC)ccn1 CC(C)C(O)CC(=O)N(C(C)C(=O)NC1CCCCCC1F)C C12CC3CC1N(C3)C(=O)C1(CCC1)C(=O)N2.c1(C2(CF)CC2)ccc(O)cc1 C1(C(=O)NCC2(NC(C(C=CCCC)O)=O)CCC2)CCS(=O)(=O)C1 [N-]=[N+]=NCC(O)CN1CCN(C2CCCCC2O)CC1 CCC(C)C(C(=O)N1C2C=CC(C2)C1COC)NC(=O)C(C1CC1)OC c1(CC(C)C(=O)NCC(O)CN(C)C(C2(c3ccno3)CC2)=O)ccc(Cl)cc1 C(CCC[Si](C)(C)C)NC(=O)C(c1ncc(Br)cc1C)N(C(CC)C)CCOC c1(C(=O)NC(C2CN(C(=O)C3=CCC3)CCO2)C)cc2c(F)c(Cl)ccc2[nH]1 C(CCCC(C)NC(=O)C(F)(F)C1CCCC1)NC(=O)CC1(CSC2CC2)CC1 c1(C(=O)OCC(=C)C)ccc(CN2CCOCC2)cc1.c12ccc(s1)CC(=O)N2 C1(NC(C(C(C)C)OC)=O)CC=C(C(=O)NCC(=O)N(C)O)C1 C1(NC(C(C)O)=O)CCCCCN(C(c2ccn(-c3cccc(Cl)c3)n2)=O)C1 N1(C(Cc2nnc(C)o2)=O)CCC2CN(C(=O)CC3CCC3(F)F)CC12 n1(CC)cc2ccc(C(=O)NCC3CCC3NC(=O)C(CC)OC)cc2n1 c1(OC)ccc(F)c(C(=O)N(C(C)CNC(C2(C)CC2Br)=O)C)c1 N1(C(c2cnn(C)c2Cl)=O)CCc2cc(-c3cn(CC(C)(C)O)nn3)ccc2C1 Cc1cc(S(N)(=O)=O)sc1C(N1CC2CCC(C1)N2C(C1(CO)CC1(F)F)=O)=O c1(CN2C(C(=O)NC(c3cccc(Br)c3)CO)CC2)cc(Br)cc(Br)c1F C#CCC(O)C(=O)NCCC1(O)CN(C(=O)C(C)(C)C2CCCC2)C1 C1(C(N2CC(N(C(C=Cc3nnc(C(C)C)o3)=O)C3CC3)C2)=O)OCCOC1(C)C CCC(C(=O)NCCCC1(NC(=O)Cc2nc(C)sc2C)CC1)C(F)(F)F N1(C(C2(CC#C)CCCCC2)=O)CCN(C(=O)Cc2ccccc2C)C(CC)C1 c1(C(N2CCCC(NC(CNC(CC)=O)=O)C2C)=O)ccc2c(c1)CC(=O)N2 C(c1ccc(F)cc1Cl)=CC(N1CCC(=CCNC(c2coc(Cl)n2)=O)CC1)=O N1(C(C(C=C)(C)CC)=O)CC2CCC1CN2C(=O)C=C(C)CCC N1(C(=O)CN(C(=O)C=CC2CCOC2)C2CCC2)CCCC(n2cccn2)C1 Cc1cc(C(=O)NC(C)C(CO)NC(c2cc(O)n(C)n2)=O)cn1C c1(C(=O)OC)nc(=NCC(C)(C)NC(=O)C=Cc2ccccc2C)cc[nH]1 N1(CC(=O)N(C(CC)C)CC)CCN(C(=O)CC(C)n2ccnc2)CC1 c1(CNC(C(C)CC(F)F)=O)cccc2c1CN(C(C1CC1C1(C)COC1)=O)C2 c1(C(=O)NCC2C(NC(CC3(COC)CC3)=O)C2)ccc(OCC(F)F)cc1 c1(CC(C(=O)N2CC(NC(C(C)SCC)=O)C2)NC(N)=O)ccc(C)cc1 CCCC(C(=O)NC1CCCN(C(c2cc(F)cc(F)c2F)=O)C1)C(C)C C1(CNS(CC=C)(=O)=O)CC2(CCN(C(=O)C=CC3CCCC3)CC2)C1 C(=O)(CS(=O)(=O)c1ccccc1)N1C2(CN(C(=O)NC(C(=O)OC)C)C2)CCC1 N1(C(C=Cc2ncn(C)c2)=O)C2CCC1CN(C(c1cocn1)=O)C2 c1(NC(=O)CC2CCC23CCC3)cccc2c1OCCC2 N1(C(C(C2CN(C(=O)OCC)C2)NC(C)=O)=O)CCC2(CC1)C(=O)NC(=O)N2C Cc1sc(O)nc1C(N1CC(=C(F)CNC(C2CC2c2ccccc2)=O)C1)=O CC1(C)CC2(CC(C(=O)NC3CN(C(c4coc(CO)c4)=O)CC3C3CC3)C2)C1 C1(CCC)CN(C(c2cccc(OC)c2)=O)CCN1C(c1ccc(OC)nn1)=O c1(C(c2n(CCC)nnn2)NCCC(c2ccccc2)C)nc(F)ccc1Br c1(CCN(CC(=O)NC2CC(CNC(C3CC3(Cl)Cl)=O)C2)C)ccccc1 C1(C)(NC(c2n(-c3cccc(OC)c3)nnn2)C(C)(C)SC)CCCCCC1 CC(C)C(F)(F)CC(=O)NC(C)C(C)NC(c1cc(Br)c(O)cc1F)=O C1(NC(c2n(CC)c(O)nc2)=O)CC2CC1N(C(=O)CCc1cccc(O)c1)C2 CC1C(c2ccccc2)CCN1C(=O)NOCC(Cl)C(C)(F)F.C1(C)CCCC1(C)C Cc1[nH]c(C)c(C(N2CCOC(C(=O)N(CCO)CCN(C)C)C2)=O)c1C C(CCN=C(NCn1ccnn1)N(C)Cc1ccoc1C)OCC C12(C(N(CC(C(=O)OC)C)C)=O)CC1CN(C(C1CCC(C)(C)C1)=O)C2 CC(C)(CCC(=O)NCC1CCCCN1C(=O)C(F)n1ccnc1)[N+](=O)[O-] N1(CC)N=C(C(=O)N(C)CCOCCN(C(=O)CC(CC)C(F)F)C)CCC1=O CC1CC(=O)NC1C(=O)NCC1(C)CCN(C(=O)C(F)(F)c2nccn2C)C1 C1(C(N(C2CN(C)C2)C)=O)CC12CN(C(=O)Nc1cccc(Cl)c1)C2 C1(NC(C2(C)CC=CC2)=O)CN(C(=O)C(C)(C)c2ccccn2)CC2(CC2)C1 C1(CC)CN(C(C2C3C=CC(C3)C2c2ccccc2)=O)CCC1O N1(c2nnc(C)o2)CCC2(CCCC2NC(c2cccnn2)=O)CC1 C1(C)(NC(c2ccc(C)nc2)=O)CCCN(C(=O)CCCc2ncco2)C1 C(=O)(C(CO)C(C)(C)C)N1C(CC(=O)NC(CC)Cn2cncn2)C2CCCC21 C1(C(=O)NC2C=CC(CC(NOCC=C)=O)C2)CCC2(CC1)CC2 C(C(C)(CNc1cc(-c2ccccc2)ccn1)CO)OC C1(NC(CCC=C)=O)CCC(COC)CC1.C12CC(C1)C(=O)N2 Cn1nccc(C(N2CC3CC(NC(C4(Cl)CC4)=O)C2C3)=O)c1=O Cc1nc(=NC(C)c2c(F)ccc3ccccc23)[nH]c2ccccc12 C1(CC)C(=O)NCCN1C(=O)C(CN=[N+]=[N-])NC(c1cnc(C)o1)=O c1(SCCCC(=O)NC2C(NC(CCCOC(C)C)=O)CCC2)ccc(Cl)cc1 CC1(CNC(=O)CC2CC2)CCN(C(C2CC(=O)N(c3ccccc3Cl)C2)=O)C1 N1(C(CC2(OC)CCC2)=O)CC2(C1)CN(C(=O)CSCc1cccc[n+]1[O-])C2 CC1CN(C(=O)CCC2CCCO2)CC1NC(=O)CCCn1ccccc1=O N1(CCCC)CCN(C(=O)C(Cc2cn[nH]c2)NC(c2ncn(C)n2)=O)CC1 C1(N(C(=O)Cc2cc(C)ns2)CCC)CCN(C(c2ccn(C)c2C)=O)CC1 c1(C(N2CCC(C(C)NC(C3C4COCC34)=O)C2)=O)ccc(O)cc1F N1(C(c2scc(C(C)=O)c2)=O)CC(CNC(c2ncccc2C(F)F)=O)CC1C Cn1[nH]c(=NC(=O)NC2CC3CCSCC3C2)c2c1CCOC2 c1(C(N(CC)CC2CCCN2C(c2cnns2)=O)=O)cnn2c1NCC(C)C2 C(C1=NOC2CN(C(C3C4CC5C(C4)C35)=O)CC12)NC(Cc1cccc(C)c1)=O c1(CNC(=O)NCc2ccnc(OC)n2)cccn(O)c1=O N1(C(c2c(C)oc(C(C)C)c2)=O)CCC(C2CCN(C(c3ccccn3)=O)C2)C1 C1(NC(c2c(C)nc[nH]2)=O)CC(CNC(=O)Cc2cccn2C)C12CCC2 CS(=O)(=O)c1ccsc1C(N1CC(C2(NC(C3CCCN3N=O)=O)CC2)C1)=O N1(C(=O)CCN(C(c2ccncc2F)=O)C2CC2)CC2CCC1CC2 Cc1cc(OCc2cscc2C)ccn1 c1(NC(C2(F)CCN(C(c3cc(Br)ccc3F)=O)C2)=O)cc(Br)ccc1CO Cc1ccc2c(c1)CCC(C(=O)NC1CC(C)N(C(C3CC3C)=O)C1)O2 C1(c2ccccc2)(NC(C(C)O)=O)CN(C(C2CC(O)(C(F)(F)F)C2)=O)C1 CCC(C)C(O)CNC(=O)CC1CCCC1NC(C1CC2(CC2)C1)=O c1(C(CC(=O)NC(CNC(C(C)C)=O)C2CC2)C)ccc(F)cc1 C1(CC(=O)NCCCCn2cccn2)CN(C(=O)C2=CCSC2)C2(CCC2)C1 c1(C(N2CCC(CN(C(CC(CC)SC)=O)C)C2)=O)cc2cc(OC)ccc2[nH]1 c1(C(=O)NCC2OCC(CNC(c3[nH]cc(C)c3)=O)C2)cccc(F)c1C#N C(C1CCC(C)CC1)=C(C(=O)NC1C(CC)CN(C(C2(C)CCC(=O)C2)=O)C1)C CC(C)C(F)C(=O)NC1(CNC(=O)C(C)SS(C)(=O)=O)CCCCC1.C(=O)(C1CC1)N C1(N(C(=O)Cc2cccnc2)CC)CCN(C(=O)Cc2nocc2C)CC1 c1(C(=O)NCC(C)O)cc(O)nc(O)n1.C1(CCOC)(C(=O)NCCN)CC1 N1(C(=O)OC)CCN(C(C2C3COCC23)=O)CC(CO)C1 CC1(NC(=O)CC23CCC2CN(C(c2ccc(I)cc2F)=O)C3)CCS(=O)(=O)C1 c1(C(N(CCC)CCNC(c2csc(C)n2)=O)=O)cccc(-n2nccn2)c1 C1(CNC(C2(O)CC(C)(C)C2)=O)CC12CCN(C(c1cccnn1)=O)CC2 C(=O)(CCC(=O)C(C)(C)C)NCC(C)CC(=O)N(CC(=O)NC1CC1)C C#CCC(CC(F)F)C(=O)NC(C)CC(=O)NC1(CCO)CCC1 c1(CC)ncc(C(=O)NC2CCN(C(C3CCCC(=O)N3)=O)CC2F)c(C)n1 C1(O)(CN(C(C=CC(CC)=CC)=O)C)CCCN(C(c2snnc2CC)=O)C1 N1(C(C2CN(c3n(C)nnn3)C2)=O)CCCC2(CC(NC(C3CC=CCC3)=O)C2)C1 CC(=O)CCCC(C)C(=O)N1CCC(CCC(=O)NC23CCN(CC2)C3)CC1 CCCC(C)(N)C(=O)N1C(C(=O)O)CCC12CC2 Cc1cnc(C(=O)NCC(CNC(=O)CCN2CCN(C)CC2)CO)cc1C#N c1(C(=O)NCCN(C(C2CC(S(C)(=O)=O)C2)=O)CC)ccc2c(c1)CCCC2 c1(C(N2C(CN(C(COCC=C)=O)C3CC3)CCC2)=O)cc(F)cc(N)c1F C1(NC(c2ccc(CCCCC)o2)=O)CCCC1(C)CNC(=O)CC(C)N(C)C N1(C(CC(C)(C)CNC(=O)NC(C)(C)C)=O)Cc2ccccc2C1 Cc1cc(C(N2CC(CNC(C3(C)CC3F)=O)C2)=O)cc(C)c1Cl N1(CCNC2CCN(C(C3CC34CCOC4)=O)C2)C(=O)NC2(CCC2)C1=O c1(C(N2CC(C)(NC(C(CC=C)C)=O)C2)=O)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] CCC(CCC(=O)NCC1CSCCN1C(=O)COCCOCCO)OC CC(C)CC(C)CC(=O)N(C1CCN(C(=O)C=Cc2ccncc2)C1)C N1(C(CCOCC#C)=O)CCC(c2nc(OC)no2)C1.C(=O)(C(C)(OCC)OC)NC C1(CC(=O)NC(CCNC(C2N(S(CC)(=O)=O)CCC2)=O)(C)C)CCCCCC1 c1(N(C(c2cccnc2)C)C)nc(NCCC2CCOC2)c2ncsc2n1 C1(F)(C(=O)NC(C(C2CC2)OC)C)CC2CCC1CC2 C#CC1(CNC(=O)C(C2CCOC2)NC(=O)C=CC(C)C)CCOCC1 C(=O)(CCCCC(N)=O)N1CC(C(C)NC(c2ccc(C3CC3)cc2Cl)=O)C1 C(=O)(C#CC(C)(C)CNC(=O)C(CC)CC=CC)NC(CCC=C)(C)C c1(C(N2CC(CCNC(c3cc(CF)on3)=O)C2)=O)nncn1-c1ccccc1 C1(N(C(=O)CCC2(C)CC2)C)CCN(C(c2cc(C(F)F)nn2C)=O)CC12CC2 N1(C(=O)CC2CS(=O)(=O)C2)CCN(C(=O)Cn2ncccc2=O)C(C2CC2)C1 c1(C(N2C(CNC(C(CC)N(C)C)=O)C=CC2)=O)ncc(OC)nc1OC N1(C(c2cccc(OC)c2OC)=O)CC2CC(NC(C3CC(OC)C3)=O)CC2C1 C=C=CC(C)C(=O)NCC1(NC(C2(O)CCOC2)=O)CC(F)(F)C1 Cc1ccc(N)cc1C(=O)NCCCNC(C1C2CCC12)=O CCCC(O)CC(=O)NC1CCCC1CNC(C1CC(C)CC(C)C1)=O C1(CNC(Cc2ccc(C)cc2)=O)CN(C(C2(F)CC=CCC2)=O)CC12CC2 C(=O)(CCC(=O)NC1CCC(CNC(c2cc[nH]c(=N)c2)=O)CC1)N(C(C)C)C CC1CN(CCc2cccc(-n3cc(C4(C)CCCN4C)nn3)c2)CCN(C)C1 C1(C)(C(=O)NC(COC)(C)C)CN(C(=O)CSc2nc[nH]n2)C1 c12cccc(C)c1c1cncnc1c(=O)[nH]2.C1(SCC)CN(C(=O)NC)CCO1 Cc1nc(C)c(C(=O)NCCN(C(c2csnc2Cl)=O)C(C)C)s1 N1(C(Cc2nc(C)on2)=O)CCN(C(c2ccc(C(NC(C)C)OC)o2)=O)C2CC12 c1(C(=O)NC(COCC)C(=O)N2CCC2C2CCCC2)ccc(C)cc1F C=CCC(CC=C)C(=O)N(C)CC1CCCN(C(=O)CCCCCCC)C1 C1(C)(C(N2CC(N(C)CC)C2)=O)CCN(C(c2cccc(CO)c2)=O)CC1 C1(C(N2CCC(C(C)NC(C3CCCS3)=O)CC2)=O)CCC2C(C1)C2(F)F N1(C(Cc2cccc(-c3ccc(C#N)cc3)n2)=O)CCC(O)C(F)(F)C1.C(C=O)O N1(C(Cc2cncc(C)c2)=O)CC(C(=O)NCC(C)(C)C)C(C)(C)C1 CCCC(O)C(CO)NC(=O)NCCc1ccc(O)cc1C CC(C)CC(C)(C)NC(=O)C(CO)NC(C1CC2CCC2C1)=O C(=O)(C(Cc1ccco1)NC(=O)NC(C)(C)CCF)OC(C)C CC(C)(C)CCC(=O)N1CCCCCC1CNC(=O)CCc1ncc[nH]1 c12cnc(s1)C2.C(=O)(C)NC(C1CN(C(C2CC2C(F)F)=O)C1)C CCC(CC)CCCC(=O)NCC1(O)CC(CNC(c2cnn[nH]2)=O)C1 C(=O)(C1=NOC2(CCOC2)C1)NCCCC(C)NC(c1c(F)cncc1Cl)=O N1(C(c2cccc(CSC)c2)=O)CCCC2(CNC(=O)CC(=O)N(C)C)CC12 C1(NC(C(COC(C)C)NC(C)=O)=O)C2CCC1N(C(=O)Cc1cnnn1C)C2 Cc1nc(C(=O)NS(=O)(=O)Cc2ccccc2)c(=O)[nH]c1C Cc1ccc(CCC(=O)NC(CCNC(=O)CC2OCCC2C)C(C)C)cc1C C(=O)(C(C)(C)F)N(CCC(C)NC(=O)CCCC1CCOCC1)C C(CCCCCCNC(C1(C)CC2CCC1C2)=O)n1cc(CNC(C)=O)nn1 C(=O)(CC(COC)COC)NC(CNC(c1cc(CC)ncc1)=O)C(C)(C)C N1(C(C2CC(=O)N2)=O)CCC2(CCCN(C(=O)C=CC3CCOCC3)C2)C1 c1(C(=O)NCCCCCN(C(c2nccc(C)n2)=O)C)cc2ccccn2c1 c1(Nc2scc(NC(=O)Nc3ncn(C)c3)n2)nnc2c(c1C#N)CCCC2 c1(-c2ccc(C(=O)Nc3c(F)ccc(C)n3)nc2)ccc(O)c(F)c1 c1(C(=O)NCC2C(C)CCN2C(=O)COCP(C)(C)=O)cc(O)nc(Cl)c1 N1(C(CCOC2CN(C(C)=O)C2)=O)CC2(CC(NC(C3COCCO3)=O)CO2)C1 CC1(C)CC(CNC(=O)C=CC2CCCN2C(c2ccc(O)cn2)=O)CO1 c1(C(=O)NCC(C)(O)CNC(=O)Cc2ccco2)c[nH]c2ccncc12 N1(C(c2c(C)nc(C(F)(F)F)s2)=O)CCC(C)(NC(C2CC(C)(C)CO2)=O)CC1 C1(CNC(=O)C=Cc2cncnc2O)CN(C(c2occc2CO)=O)CC1(F)CO N1(C(C(C)SCc2ccccc2)=O)CCC(O)(CN(C(=O)C=CCF)C)CC1 C(=O)(C(C)S(N)(=O)=O)NCC1C(NC(C2CCN(CCC#C)CC2)=O)CC1 N1(C(CCN(C)C(c2cc(C3CC3)nn2C)=O)=O)CCC2(CCOC2)C1 C1(CC)C(C(=O)NC2CC2C(C)C)CCCN1C(C1CCCCC1(C)C)=O CC(C(CO)NC(=O)CCNC(C1CCCO1)=O)NC(=O)COC1(C)CCCC1 C(CC(F)(F)Cn1cc(C2(O)CCOCC2)nn1)NC(C(C)OC1CCOC1)=O C12CN(C3CC13)C(=O)N2.C(=O)(CC(=O)NC(=O)COc1ccccc1)OCC.OCC N1(C(c2c(C)ncc([N+](=O)[O-])c2)=O)CCCC(C2CN(C(C3CC3F)=O)C2)C1 C1(C(N(C(C(CC)C)C)C2CC2)=O)CCN(C(=O)c2ccc(N)cn2)O1 c1(NCC2C(C)CN(C(=O)C3=NNC(C(F)(F)F)C3)C2)c[nH]nc1S(N)(=O)=O c1(C(=O)NCC(C)NC(=O)Cc2csnn2)nnn2c1CCC2 CN1CCCCC1C(=O)NCCC1CCCN1C(=O)CC1C(C)(C)C1(C)C C1(C(C)(C)NC(c2cocn2)=O)CCN(C(=O)Cc2cccc(F)c2)CC1 c1(OC2CC(NC(=O)OC(C)(C)C)CC2O)cc(Cc2nn[nH]n2)ccc1F N1(C(C2CC(C)OC(C)C2)=O)CC2(CCCC2NC(c2ncccc2N)=O)C1 C1(Cl)(C(=O)NCCC(C)N(C)C(C2CC(C(F)F)C2)=O)CC1(F)F C(C(=O)N1CCC(C(=O)NCC2(C(N)=O)CC2)(COC)C1)(C(C)C)OCC N1(C(C=C(C)CNC(c2cnn3cccc3c2)=O)=O)CCN(C)C2(CC2)C1 C(C(F)(F)C(F)(F)F)OCC(=O)NC(CN(C(C1C(=C)C1)=O)C)C C1(C(N(CCn2c(C)ncc2)C)=O)CCCCN1C(=O)Cc1cncn1C C1(CNC(c2cnccc2C(F)(F)F)=O)COCCN1C(C1CCC2CC2C1)=O C1(C(=O)NCc2nc(CNC(C3(C(C)C)CC3)=O)sc2)CC2C=CC1C2 N1(C(c2ccc(CSC)cc2)=O)CCCCC(CNC(=O)CNS(C)(=O)=O)C1 c1(C(N2CCC(N(C(CNC=O)=O)CCO)C2)=O)nccc2c(Cl)cccc12 C1(NC(=O)NCC(C)OC)CCN(c2ccc(C(F)(F)F)cn2)CC1 c1(C(=O)NC(CNC(=O)C2=CC(O)CCC2)CO)ccc2cnccc2n1 C(=O)(CCCC(C)C)Nc1occ(C(N(CC(COC)O)C)=O)n1 c1(C(N2CCC(NC(C3C(C)(C)OCC3)=O)(CO)CC2)=O)cc(S(C)(=O)=O)co1 C(=O)(CCCS(C)(=O)=O)N1CC(C)(C)C(CNC(=O)C(F)CC2CCCC2)C1 c1(C(=O)NC2CCCC2NC(c2n[nH]cc2Cl)=O)ccc2c(c1)CCC(O)C2 N1(C(C(C2CCCCCC2)C)=O)CCC(C(=O)NCc2cc[nH]c(=N)c2)C(O)C1 N1(C(C(CC)O)=O)CCC(C)(CNC(c2ccc(COC)c(F)c2)=O)CC1 C1(NC(c2c(C)cc(CC)o2)=O)CCC(C)N(C(=O)Cc2ccc(C)cc2C)C1 c1(C(=O)OCC2OCCCN(S(CCOCC)(=O)=O)C2)c(Br)cc(Br)c(O)c1Br c1(N(C(CNC(C(C)OCCOC2CCCO2)=O)C)C)nccn1C.OC N1(C(c2cn(C)nc2)C(=O)NCCOCC2CC2)CC2C(C1)C2(F)F c1(CCNC(C2CC(=C)C2)=O)nccc(N(CCOC(C)=O)C(C)C)n1 Cc1nn(C2CC2)cc1C(=O)NCC1CCCN(C(C2CC(F)(CO)C2)=O)C1 C1(C(N(C(=O)NC(C(C)C)CN(C)C)C2CC2)=O)CCCOC1c1ccccc1 C(=O)(CCC(C)(C)C)NCC(CC)NC(c1c(C)nn(C)c1OC)=O C(=O)(CC(C)C(F)(F)F)NCCCCC1CN(C(c2c(C)nc[nH]2)=O)C1 CCCCCC(N=c1cc(C)nc(C2CCCO2)[nH]1)c1ccco1 c1(C(=O)NCC(c2ccccc2)NC(=O)CCF)ccc(F)c(F)c1 CN1CCCCC1C(=O)N(C(C(=O)NCCCCCN=[N+]=[N-])C1CC1)C C1(NC(C=C(CC)C)=O)CC12CCC(NC(C1CCC3(CCC3)O1)=O)CC2 N1(C(CC=CC=C)=O)CC2CC1(C(N1C(CO)CC1CO)=O)C2 c1(C(=O)NC2CCN(C(c3c(C)coc3)=O)C(C)C2)cc(F)c(N)c(F)c1 C1(C(N2CC3(C(NC(c4ccc(C5CC5)s4)=O)CC3)C2)=O)CCC2(CCC2)O1 C#Cc1ccc(C(=O)NC(c2ccnn2C)C(=O)NCc2ocnc2C)o1 c1(CC(=O)NCC(CO)NC(C2C(OCC)C2)=O)ccc2c(c1)CCCC2 N1(C(c2nc(C)oc2)=O)CCCC12CCCN(C(=O)CCC(C)N(C)C)C2 Cc1cc(C(=O)NCC2CN(C(=O)CCF)CC2C(F)(F)F)c(O)nn1 c1(C(N2C3CCC2CN(C(C2(F)CCC(F)(F)C2)=O)C3)=O)c(F)cc(F)cc1Cl n1(N2CCCC2)cnc2c(N3CCCC(SCC)C3)[nH]c(=NCC3C=CCC3)nc12 N1(C(CNC(=O)OC)=O)CCCC1.C12CC(C1)C(=O)N2.C(F)(F)(CC)C1(C)CC1 C=C1CC(CC(=O)NCCCOCCC(=O)NCCn2cncn2)C1 C1(C(=O)NCC2C(C)(C)CCN2)CCNCC2(CC2)C1 C1(CCC)CCC(C(=O)NC23CC(NC(C4(C#N)CC4(C)C)=O)(C2)C3)CC1 Cc1cc(C(N2CCNC(=O)C2c2ccccc2)C(=O)NCCC#N)cc(C)n1 n1(CC(=O)NNC(c2ccc3c(O)n[nH]c3c2)=O)nc2n(c1=O)CCCCC2 CC1(C(=O)NCCCCO)CCN(C(=O)CCCc2ccc(Br)cc2)C1 C(=O)(C(C)(C)CF)N1CCC(C(C)NC(=O)COCc2ccccc2)C1 c1(CNC(C(c2cccs2)N(CCC)CC)=O)ccccc1Br C1(C(N2CC(C)N(C(=O)CC#N)CC2)=O)CCc2cnn(C)c2C1 C(C)(C)(C(C)CC(=O)NC(c1cccs1)CO)NC(c1c(CC)cccc1)=O C(=O)(C1=C(F)CN(C(=O)C(C)SC(C)C)CC1)NC(CCC=C)C1CC1 C#CCC(CC(=O)NC1CNC(=O)C1(C)C)NC(=O)C=CC(=O)N(C)C CC1=Nc2ccc(C(=O)NCC3CC=CCO3)cc2C1(C)C C1(NC(C(CO)NC(N)=O)=O)CCCN(C(=O)COc2ccccc2)C1 C(CO)(CCCNC(C1CC2C=CC1C2)=O)NC(Cc1ccc(C(C)=O)s1)=O C#CCC(C)(C(=O)Nc1nc[nH]n1)NC(=O)CSCC(C)(C)COC n12c3c(cc(cc3)c1=O)CC2.c1(C(N2CCN(OC(C)=O)C2)=O)ccncc1O N1(C(CN(CC)CC)=O)CCC(CC(C)NC(c2cnsc2)=O)CC1 c1(CS(C)(=O)=O)ccc(-c2nc(COC(F)(F)F)no2)cc1 CCCC(C)(C)CC(=O)NCCCN(C1CCCC1)C(c1ccc(F)c(O)c1)=O C1(C(=O)NCc2cc(C)no2)C2CCC(C2)N1C(c1cc(=O)cc[nH]1)=O N1(C(c2cc(=NC)[nH]cc2)=O)CCC2CN(C(=O)CSC(F)F)C2C1 C(=O)(C1=CC(O)C(NC(C2CN3CCN2CC3)=O)C1)N1CC(CC(C)C)OCC1 c1(N2CCN(C)C3(C2)CCOC3)nc(=NC2CCC(O)C2)[nH]c2ccccc12 C1(NC(C(C)n2cncn2)=O)CCCC1(F)F.C12CC1CN(C)C2=O C#Cc1ccc(C(=O)NC(C)C(C)(C)NC(=O)Cc2nocc2C)c(F)c1 c1(C(=O)NC2(CNC(C(C)(C)C3CCCO3)=O)CC2)ncccc1F c1(C(N(CCN(C(=O)CN2CC3CCC2C3)CC)CC)=O)cc(F)ccc1F CCC(F)(F)C(C)(C)C(=O)NC1CN(C(=O)COCC2CCCO2)CCC1CO C1(C(=O)NCC23CC(NC(COCCC)=O)(C2)C3)CC2(C1)CS(=O)(=O)C2 C1(C(=O)NC(CCOC)C)CN(C(c2cncc(OC)c2)=O)CCO1 Cc1cc(F)c(C(=O)N(C)CCOCCCSc2ccc(S(C)=O)cc2)cc1F c1(NC(CC)=O)ccc(C(=O)NC2CCCCC2C)cc1 c1(CC(=O)NCCC(=C)CNC(=O)CSc2cccc(Cl)c2)c[nH]ccc1=O C1(N(C(C2(CC(=O)CC3COCC(C)O3)CCCO2)=O)CC)CCCCCC1O CC1COCC(C(=O)NC(C2(C(N3CCC(F)(CO)C3)=O)CC2)C)O1 CC1C(C(=O)NC2COC(C(F)F)C2)CCN1C(=O)C1=CCCC1 c1(CC(=O)NC2CCC(CNC(=O)CCCF)CC2)ccc(Cl)cc1 C1(NC(C(CC)C(C)O)=O)CCCCC12CCCN(C(=O)C(CC)CCOC)C2 N1(S(CC=C)(=O)=O)CCC2(CC1)CNC(=O)C2.c12cnc(s1)NC1CN(C1)C2=O c1(C(=O)NCC2(C)CCN(C(=O)C(O)CF)C2)ccnc2ccnn12 C(C(=O)Nc1cccc(CC2CC2)c1)(C(Cc1ccccc1)OC)NC(=O)OC C=CC(C)(C)CC(=O)N1CCN(C(C)=O)C(OC(F)F)C1 N12CC3CC1C3C2=O.c1(C(=O)NC2C(NC(=O)OCC)CC2)cc(C2CC2)on1 CC(C)C(O)CC(=O)NCCN(C(C1CCCN1C(=O)NC)=O)Cc1ccsc1 C(=O)(CCC(C)(C)C)NCC1(C(C)NC(C2CC(c3ccccc3)C2)=O)CC1 C1(C(=O)NCC(C)NC(c2cccc(CS(C)=O)c2)=O)CN(C)CCN(C)C1 C1(NC(C(Cn2cncn2)NC(C2(CC=C)CCCC2)=O)=O)CC12CCCCC2 N1(C(c2cnc(CC)s2)=O)C2CCC1CC(N(C)C(c1cccc(F)c1F)=O)C2 C1(C(N(C)Cc2ccccc2)=O)COCCN1C(=O)Cc1cc[nH]c1 c1(SC)nc(N2CCC(n3cc(COC)nn3)C(O)C2)ncc1C c1(N(C(C=C)COC)C)nc(=NCC(C)c2ccsc2)[nH]c2ccccc12 C1(C(N(CC(C(=O)N(CC(C)N(C(C)=O)C)C)C)C)=O)CCC2(CC2)C1 Cc1cccnc1CCC(=O)NCC1CCCN(C(C2(Cl)CC2)=O)C1 N1(C(c2n(CC)ncn2)=O)CC2(CCC(CNC(C3C=CC3C(=O)OC)=O)O2)C1 Cc1cccnc1C(=O)NCC(C)NC(c1ccccc1-c1ccncc1)=O CC(C)CCCCC(=O)N1CC(CCNC(c2ccc(Cl)[nH]2)=O)C(C)C1 c1(OCCCC)ccc(NCc2ccc(I)c3nsnc23)cc1OCC N1(C(Cn2c(C(C)C)ncc2)=O)CCC(C)C(NC(C2CC2C(C)O)=O)C1 C(C(=O)NCC(F)CNC(c1ccc(CO)s1)=O)(C(C)C)NC(C)=O Cc1c(C(=O)NCCN(C)C(c2occc2F)=O)nn2c1CCCC2 C1(C(C)NC(C2(C(F)F)CCCC2)=O)CCCN(C(=O)C(C)(C)C#N)C1 C1(O)(CNC(CCC=C)=O)CCN(C(C2OCCCC2c2ccccc2)=O)CC1 N1(C(c2cccc(F)c2O)=O)CC2(CCCN2C(=O)CCC2CC2)C1 N1(CCCCNC(C(CC)O)=O)CCCC(CN(C)C)C1 N1(C(C(CC2CC2)OC)=O)C2CC1CN(C(c1cc(O)cc(F)c1)=O)C2 N1(c2n(CCC#C)c(C(c3ncccc3F)C)nn2)CCNC(=O)C1C CC1C2CC(C2NC(=O)C2=CCCCC2)N1C(c1cnoc1-c1cccs1)=O Cc1cc(C(N2CCN(C(=O)C(C)(C)F)CC2CC2CC2)=O)nnc1C CC(O)CCCc1cn(CC2CCNC2)nn1 CCCCC(CNC(=O)CSc1cn[nH]c1)NC(C1(C)CC=CCC1)=O Cc1nc2c(o1)CCCC2CC(=O)N1CC(NC(=O)C2=COCCO2)CC(C)C1 c1(C(=O)NC2CN(C(C3CCN(CC#C)CC3)=O)C2)ccc(SC)cc1C c1(C(N2C(C(N(C)Cc3ccc(C)cc3)=O)CC(F)C2)=O)cccc(I)c1F Nc1cc(F)cc(Cl)c1C(N1CCN(C(c2cccc(=O)o2)=O)C(CO)C1)=O Cc1ccc(C(=O)NC2CCC(CNC(=O)Cc3[nH]cnc3C)C2)cc1 c1(C(N(CC(C)NC(C(CC)(C)C(N)=O)=O)C)=O)cc(=O)c2ccccc2[nH]1 C(=O)(C(C(C)(C)C)C1CCC1)N(C1CCN(C(c2cc(OC)nn2C)=O)C1)C N1(C(CC=C)=O)CC2CC(NC(c3cccnc3C(F)F)=O)C(C2)C1 C1(NC(c2c[nH]c(=N)s2)=O)CCN(CCNC(C2CC(n3ccnn3)C2)=O)CC1 N1(C(=O)Cc2cnsc2)CCC2(C1)CN(C(C1CC13CCCOC3)=O)C2 c1(C(N2CC(N(C(CN3CCCC(CC)C3)=O)C)C2)=O)ccc(F)cc1C(F)F C12(C(=O)NCC3CCCCN3C)CC(CO)(CN1C(=O)CCCn1ccnc1)C2 C1(CNC(C(CC)F)=O)CN(C(C2(COC)CC(F)(F)C2)=O)CCCO1 CC(O)CC(C(=O)O)NC(C1CCCCC1C)=O N1(CCNC(CN(C(CC=C(C)C)=O)C)=O)CCCC1C(C)O C1(OCC)CN(C(c2ccsn2)=O)CC1CNC(c1ccccc1COC)=O c1(OCC(NNC(c2ccc(C#C)cc2)=O)=O)ccc2c(c1)CCC2 N1(C(CC2CNC(=O)O2)=O)CCCC12CCCN(C(=O)C1CC1)C2 C(C(C)C)(C(O)C(=O)N1CCN(C(c2ccc(=N)[nH]c2)=O)C(CO)C1)OC N1(C(c2c(C)[nH]cc2)=O)CC2CC1CCN2C(=O)C(C)CC1CCCCC1 c1(C(N2CCC3(C(NC(C(C)CC4CCC4)=O)C3)C2)=O)cc(Cl)c(Cl)c(Cl)c1 C1(C(=O)NCC(C)(C)O)CCC(NC(C2CCCO2)=O)CC1 C1(N(C(=O)C(=C2CCCCC2)F)C)CN(C(=O)C(O)C2CCC2)C2(CCC2)C1 C(=O)(C(C)CCC(C)(C)C)NC1CC(C)N(C(=O)C(C)(F)F)C1 c1(CNC(C2N(C(C(C)Cn3ccnc3)=O)CC2)=O)c(Cl)cccc1Cl CC1CN(C(=O)CC2CCC2)CC1CNC(=O)CCOc1cccc(Cl)c1 c1(NCC(CC(C)C)NC(=O)Cc2cscn2)cc(Cl)nc(S(C)(=O)=O)n1 N1(C(CC(=O)NCC)=O)C2CCC1CC(O)(CNC(C1CC(O)CN1C)=O)C2 C(C(C)(C)CNC(c1cnn[nH]1)=O)N(C)C(c1ccc(C(F)(F)F)o1)=O C(CCCC(=O)NC1(CN(C)C)CC1)NC(CNC(C1C(C)C1)=O)=O.C(C)=C c1(C(=O)NCC2(C(N(CCC(C)C)C)=O)CC2)cc(OC2CC2)no1 C1(NC(c2c(C)oc(C(C)C)c2)=O)CC2(CCCN2C(=O)CC2CCOC2=O)C1 CN1C(=O)COCC1CNC(C1CC(O)CN1C(C1CC2(CCC2)C1)=O)=O Cc1cn2cc(C(N3CC4(CCCC4NC(c4cnn(C)c4F)=O)C3)=O)nc2s1 N1(C(c2c(C)n(C)cc2)=O)CCCC(C)(NC(c2sc(C(F)(F)F)nc2Cl)=O)C1 C(CNC(c1cnc(O)cc1OC)=O)(C(C)C(C)C)NC(c1c(CC)scc1)=O c1(CC(=O)NCCC2CCN(C(C3OCCCO3)=O)C2)cccc2c1OCCO2 N1(C(c2ccc(CC)s2)=O)CC(NC(=O)C(F)Cc2ccccc2)CC2(CC2)C1 Cc1cc(C(N2CC(NC(=O)CC3CCCC(C)O3)CC(O)C2)=O)c(O)nn1 CC1CC(C(=O)NCc2cccc(C(=O)NCC[Si](C)(C)C)n2)CCO1 c1(C(N(CC(C)N(C)C(C2CC(C)N(C)C2)=O)C)=O)cc(N2CCCC2)ccn1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(NC(C2CCC(CO)CC2)=O)CC(O)C1 Cc1cc(C(=O)NCCCC2CCCN2C(c2cc(Cl)n[nH]2)=O)c(O)nn1 C(=O)(C1=CCCN(CCC)C1)N1CCCC(NC(C2CCC2)=O)C1 N1(C(c2c(CC)nccn2)=O)CC2CCCC(NC(=O)Cn3cccc3)C2C1 c1(C(=O)NCC(CCNC(C(C(C)OC)N(C)C)=O)O)cccc2[nH]ccc12 C#Cc1c[nH]nc1C(=O)NCCCC(c1ccccc1)NC(=O)CSS(C)(=O)=O CCCC(C(=O)NCC1CCC=CO1)NC(C1(CC)CC(C)(C)C1)=O Cc1ccc(S(C)(=O)=O)cc1C(=O)NC1CCN(C(c2nc(Br)c[nH]2)=O)C1 Cc1cccn2nc(C(N3CCC(NC(c4ccc(F)c(Cl)c4N)=O)C3)=O)cc12 C1(C(N2CC3(CN(C(c4ccc(CC)c(F)c4)=O)C3)C2)=O)CCC2(CCC2)OC1 c1(NC)c(C(=O)NC(C)CCC(=O)Nc2ccc(CO)cc2O)cnn1C C1(OC)CC(CNC(c2nccnc2C)=O)N(C(c2cc(C)n(C)n2)=O)C1 Cc1cnc(CC(=O)NC(CNC(=O)C(F)CC2CCOC2)C2CC2)o1 C(=O)(C(C#N)C(C)C)N(CC(C)N(C(c1nccc(CC)c1)=O)C)C C1(SC)NC(=O)C(C)CN=C1NC(=O)NC(C)(C)CSC.C(C)(C)(C)O c1(C(=O)NCCCN(C(c2c(CCC)nns2)=O)C(C)C)cncc2c1CCC2 C(=O)(C#CC1(C)CCCO1)N(CC)CC1CCCN1C(=O)CC1CCCN(C)C1 c1(C(=O)NCc2cc(C(=O)NC(c3nc(C)no3)CC)sc2)cn(C)c(=O)n1C N1(C(CC(=C=C)C)=O)CCC(C2(NC(C3CCc4nnc(C)n4C3)=O)CC2)CC1 c1(CC)ccc(C(=O)NC(C)CCCCNC(=O)Cc2ncccc2C)c(C)c1 c1(C(=O)NC2CC(NC(CC(C)NC(N)=O)=O)C2)c(Cl)ccc2c[nH]nc12 c1(CNC(C(C)n2ccnn2)=O)cc(C(=O)N(CC(C)O)C2CC2)on1 N1(C(C(C)C2CC2)=O)CCC(O)(C(C)NC(=O)CCOC2CC2)C1 S(=O)(=O)(c1cnc(Cl)c(C(F)(F)F)c1)Nc1cc(Br)cc(CC)c1O c1(C(=O)NCCC(N2CC(C(C)NC(C3CC3F)=O)C2)=O)nc2ccccc2s1 N1(C(c2c(CC)nns2)=O)CCC2CC2(C(=O)NC(COC)CO)CC1 C#CCN(OC)C(=O)C1C=CC(NC(=O)CC2CCCC2)C1 CCN=C(NCc1nnc(CC)s1)NCC1CC1(F)F C1(C(N(C)CC2CCCC3CC23)=O)CCC(CNC(C2CC(C)(C)CO2)=O)CC1 CC(C)CC(CNC(C1CC12CC2)=O)NC(C1CC(F)C(=O)N1)=O N1(C(c2cnn(CCC)c2C)=O)CC(NC(=O)CP(C)(C)=O)C2(CC2)C1 c1(C(=O)NC(C(C)NC(C2CC=CC(O)C2)=O)C)c[nH]c2nccc-2c1 CC1(C)CCOC(CC(N2CC3(C(=O)NC4(CCCF)CC4)CC2CO3)=O)C1 N1(C(Cc2ncc(C)s2)=O)CCOC2(C1)CN(C(C1(C)CC3(CCC3)C1)=O)C2 N1(CC(=C)Br)CCCC(N(C(=O)CC2(C(F)(F)F)CC2)CC)C1C CC(C)C(C)(CNC(c1ccccc1-c1cncnc1)=O)NC(=O)CSCC#N N1(CC(N2CCCC(C(CC)NC(C=CC(C)C)=O)C2)=O)CC(=O)N(C)C1=O c1(C(=O)NCC2N(C(CCC(=O)OCC)=O)CCC2)ccc(C#CC2CC2)cc1 c1(C(C)C)c(N(C)CC2CCCN(C(=O)C(C)OCC3CC3)C2)ncnc1Cl C=C1CCC(C(N2C(C(=O)NCc3nnnn3C(C)C)CCC2C2CC2)=O)CC1 C1(C(=O)NC2C(C)N(C(C3CCOCC3)=O)CCC2)CCC2CCCCN12 CCC(CCC(=O)NOCCC1CC1)NC(=O)C(C)(C)n1ccnn1 C1(CNC(=O)CC2CCCCO2)CCN(C(c2cn(CCF)nn2)=O)CC1(F)F c1(C(N(CC(CN(C(=O)C(c2ccc(F)cc2)C)C)O)C)=O)ccc(N)cn1 N1(CCC(=O)NCCC(CNC(CC2CC(C)(C)C2)=O)O)CCCCC1=O C(C(C)(C(C)C)NC(=O)CCOCCN(C)C)NC(Cc1c(C)ocn1)=O C(C(C(=O)N1CCC12CCCC2)C(C)C)NC(C(COC)(F)F)=O C1(CNC(=O)CCc2nccs2)(CNC(=O)CC2(CO)CC2)CC12CCC2 C(C(C)(C)CC(=O)N(CC(C)NC(=O)C(CC)NC(N)=O)CC)CC CC1OCCN(C(C2CCC3(CC3)C2)=O)C1C(=O)NOCC1(C)CCC1 Cc1ncn(C)c(=O)c1C(=O)NCCC(C)NC(=O)Cc1ccccc1 c1(C(=O)OC(C(=O)OCC)C(C)C)ccc(NC(=O)COC)c(C)c1 C1(NC(C2C(C)(C)NC(=O)C2)=O)CCN(C(C2CCCC23CCC3)=O)CC1(C)C N1(C(C(CC)NC(N)=O)=O)CC2(CC(NC(c3cc(C(F)F)cc(C)c3)=O)C2)C1 c1(CCCC)ccc(C(=O)NC(C)CNC(=O)CCN(CCCOC)C)s1 N1(C(C2=C(C)CCC2)=O)CCC2(CCC(NC(C3CC(n4ccnc4)C3)=O)C2)C1 c1(C(N2CC(CNC(CC(CN(C)C)O)=O)C(O)C2)=O)cccc([N+](=O)[O-])c1 c1(C(N(CC(C(=O)N(CC=C)CCO)C)C)=O)ccc(F)c(O)c1 c1(C(=O)NC2(CN(C(=O)C(O)CC3CCCC3)C)CC2)sccc1C#N n1(C(C)C)cnnc1CCNC(c1nc(C2CC2)cs1)=O C(=O)(C(C)CCC(C)(C)C)NCC1N(C(c2c(C)ccs2)=O)CC(F)(F)C1 Cc1nc(C(=O)NCC2(F)CN(C(c3ccnn3C3CCCC3)=O)C2)co1 C=CCC(F)(F)CN(C)C(C1C(C)CCN1C(=O)COCCCOC)=O C1(C(N(CC(C)NC(c2cc(Br)n(C)n2)=O)CC)=O)CC2(CCC2)CO1 c1(OC)c(C(=O)NCCCCCN2CCN(C(c3cc[nH]c3)=O)CC2)csc1C C1(CN(C(c2ccn(CCC)n2)=O)CC)CCCN(C(=O)COC2CCCC2)C1 Cc1c(NCc2cc(F)cc(Br)c2)ncnc1NC1CCCC1CCC(C)C c1(CNc2n(C(C)(C)C)ncc2C(=O)O)c(Cl)ccnc1F c1(C(N2CCN(C(C3ON=C(C)C3)=O)C(CCO)C2)=O)ccc2cc(C)cn2c1 N1(C(C2C(C)(C)CCN2C(c2ccc(O)c(F)c2)=O)=O)CC2C3CCC(C3)C12 Cc1cccc(CC(N2CCC=CC2C(=O)NCC2CN(C(C)C)C2)=O)c1 CC(C)(C(=O)NCCOC1CCN(C(C2C=CCC2)=O)C1)c1cccs1 C(CCC(C)C(=O)NCCCC1CCCN1C(=O)C(C)C(C)C)OC CC(C)C(C(C)NC(=O)CCCn1c(O)nnc1O)NC(=O)C=Cc1cn(C)nn1 c1(OCCC(=O)NCC(C2CC2)NC(=O)CC2CS(=O)(=O)C2)cccc(F)c1 N1(C(c2snnc2C2CC2)=O)CCC2CCN(C(C3CCCO3)=O)C2C1 N1(C(CC2(CC)CCC2)=O)CC2CC(C)N(C(=O)C(C)c3ccco3)C2C1 n1(NC(=O)CC2CC(C)(NCC(c3ccc(O)cc3)O)C2)ncc2ccccc12 C1(CNC(c2c(C)ncn2C)=O)CN(C(=O)CSC2CCOC2=O)CCC1C c1(OC)ccc(C(N2CCCC2C(C)NC(c2occc2C)=O)=O)cc1 C1(NC(CC2OCCCN(C(C=C(C)C(C)C)=O)C2)=O)CCN(C)CC1(C)C C1(C(=O)NC(CCCC)CNC(c2nonc2N)=O)CS(=O)(=O)CC12CC2 CCC(CC(=O)NC(C)CC1CN(C(=O)Cc2cccc(C(F)(F)F)c2)C1)OC C1(C(N2CCC(C)(CNC(c3ccncc3)=O)C2)=O)COc2ccc(Cl)cc2O1 C1(NC(c2cc(C)c(C)[nH]2)=O)CC2CN(C(=O)C#CC3CC3)CCN2C1=O N1(C(CCn2ccc(C)n2)=O)CC(NC(=O)C(c2ccc(Cl)cc2)CO)C(C)C1 C(CCCC(=O)N1CC(F)CC1CC(=O)N(C(C)CCO)C)OC C1(CC)C(NC(=O)CCCN(C)C(=O)C2CC2)CCN1C(c1ocnc1C)=O Cc1sc(C(=O)NC2COCC2CNC(C2C(C)C2C)=O)cc1[N+](=O)[O-] C=CC(C)(O)CC(=O)NCC(c1ccc(OC)cc1)NC(=O)CC1CCC1 C(C)(CCC(=O)NC1CCSC1)NC(C(n1ccc(C)n1)C)=O Cc1cccc(Cl)c1NC(=O)CCn1nc(C2CC2)nc1-c1cc2sccc2s1 c1(C(=O)NC(C)Cn2cc(CN3CCCC3CO)nn2)cc2cc(Cl)ccc2o1 C#Cc1cncc(C(c2nnnn2CC=C)NCC2CC3(CC3)C(=O)O2)c1 O=C1CC(C(N2CC(C(N3CCC(CCCO)C3)=O)C2)=O)CN1 c1(C(N2CCC(NC(C(CC=CC)C)=O)C2)=O)c(N)cccc1Cl C1(C)(C(=O)NC(c2nccn2C)C)C=CCN1C(c1ccc(CO)o1)=O c1(C(CNC(CC)C(=O)N(C)C)OC)ccc(O)cc1 N#Cc1ccc(Br)c(CN2CC3CCC2CN3C(c2sccc2Cl)=O)c1 C(=O)(C(O)CC(C)C)NC1(C(=O)NC(CC)CC)CCSC1 C(=O)(C(C)C(F)(F)F)NC1C(OC)CN(C(c2[nH]cnc2C#N)=O)C1 C1(C(=O)NC2CCC(SC)CC2)CCC(C)(C)CO1.n12cc(nn1)COCC2 c1(C(N2C(CNC(c3[nH]cc(-c4[nH]c(=N)sc4)c3)=O)CC2)=O)ccccc1F c1(C(=O)NCC(C)CN(C(=O)C(=Cc2c[nH]cn2)F)C)ccn(C)c(=O)c1 N1(C(CNC(CCC)=O)=O)CCC(O)(CCNC(C2CC2CC)=O)C1 C1(C(=O)NCC(C(C)C)(C)C)CC(O)C(O)CC1CNC(c1cccnc1S)=O c1(C(=O)Nc2ccc(C(C)=O)cc2F)cc(C2=CCSCC2)cn1C C1(NC(CC=CCNC(c2c(C)ccnc2)=O)=O)CCC(C2CC2)C1 C#Cc1ccc(C)c(NC(c2cccc(COC)n2)c2nnnn2CCC)c1 c1(C(N2CCC(c3scc(C)n3)C2)=O)ncccc1Cl.c12cn(nn1)CCNC2=O C(=O)(C1=NOC2(CCN(C(=O)CC3CCC3)C2)C1)N1C(C)CC(C)(C)C1 c1(CN2C(C(=O)Nc3cncc(C)c3)CC(F)C2)cccc2ccncc12 C(CN=c1nc(N2CCC(c3cccs3)CC2)c2c(ncn2CC)[nH]1)SCCC=C c1(OC)ccc(NCC(=O)NCC(O)COc2cnccc2CBr)cc1F C1(C(N(C)Cc2cc(C)cc(F)c2)=O)N(C(c2csnn2)=O)CCCC1(C)C CC1=NOC(=O)C1CCC(=O)NCC1CCN(C(c2cc(C)n(C)c2)=O)CC1 c1(C(=O)NC2CCC(NC(c3c(OC)noc3C)=O)CC2)cnc2ccoc2c1 C12(C(N(CCCN(C(c3n(CC)ccc3)=O)C)C)=O)CCCCC1CS(=O)(=O)C2 CC(C)CC(C(=O)NCC1CC(F)C1)ONC(c1ccc(F)cn1)=O Cc1c(CNC(C2CCC(NC(=O)C(O)c3ccsc3)C2)=O)cccc1F C1(C(=O)NC2CCN(C(CC=C)=O)CCC2CO)CCc2nc(CC)ncc2C1 C1(=O)C(N)COCCN1C.C1(C2CC2)(OCC(=O)OC)CCC1.C(CC(C)C)O Cc1[nH]nc(CO)c1C(=O)N(C(c1ccccc1-c1nn[nH]n1)=O)C(C)C c1(C(N2CC(OC)(CNC(=O)C(C)(F)C(C)(C)F)C2)=O)nccn2c(C)nnc12 N1(C(C(CNC(c2c(CC)nn[nH]2)=O)OC)=O)CCc2nc(O)[nH]c2C1 N1(C(c2c(C)c(Cl)cnc2)=O)C2CCC1CC(CC(C)NC(c1cnns1)=O)C2 C#CC1(O)CCN(CCC(=O)NC(=O)C)C1.C(=O)C(C)(C)C N1(C(CCc2ncc(C)[nH]2)=O)CCCC(N(C(=O)CC2CCOC2)C)C1 Cc1cc(C(=O)NCCCC(O)C(=O)N2CCCC2(C)C(C)(C)C)c(C)nn1 N1(C(C2C(CNC(CC(C(C)C)C)=O)C2)=O)CC2(CCNC2=O)C1 C1(C(N2C(C(=O)NCC(=O)NC3CCC3)C(O)CC2)=O)CC2CCCC2C1 CC1CS(=O)CCN1C(C1CN(C(C2CCCN2C=O)=O)CC1F)=O N1(C(c2ccc(CC)nc2)=O)CCC2(CC1)CN(C(c1ccc(C)cn1)=O)C2 Cc1ncc(F)c(N2CCCC(CC(=O)Nc3ccc(Cl)cc3O)C2)n1 C12(C(N(CC(CNC(C=CCC)=O)C)C)=O)CCCC(C(=O)OC)(COC1)C2 C#Cc1cc(C(N2CCC(C(=O)NC(c3cn(C)cn3)C)C2CC)=O)ccc1C C(CC(O)C(C)C)NC(C(C1CN(C(=O)C(O)CN(C)C)C1)OC)=O c1(C(N(C(CNC(C(CC#C)C)=O)C)CC)=O)cc(Cl)cnc1C Cc1cccc(Cl)c1C(=O)NC1CC1CNC(c1coc(C2CCC2)n1)=O N1(C(C2C(C)OCC2)=O)CCCC(C2CN(C(c3ccccc3[N+](=O)[O-])=O)C2)C1 c1(CC(=O)NC(CC)(CNC(c2nsnc2O)=O)CC)ccc2c(c1)CC2 N1(C(C(CC#C)O)=O)CC23CCCC2(C1)CN(C(c1sccc1Cl)=O)C3 Cn1ccn2ncc(C(=O)NC3CC(NC(c4n[nH]c5c4COC5)=O)C(O)C3)c12 C12(CNC(Cc3c(C)cco3)=O)CC(CO1)N(C(=O)CC1C=NN(C)C1=O)C2 C(=O)(C(F)(CNC(C1(CO)CCCCO1)=O)C(C)C)N1CCN(CCOC)CC1 C1(NC(C(CC)N(CC)CC)=O)CN(C(=O)Cc2cccs2)CCC1(C)C N1(Cc2c(C)csc2)CC(O)CC1C(=O)Nc1cc(O)n[nH]1 N1(C(C)C)CCOC(CN2CCC(N(C(=O)Cc3coc(C(F)F)n3)C)C2)C1 N1(C(C(C=C)O)=O)CCCC2(C1)CN(C(=O)CC(C)c1ccccc1)C2 C1(CNC(Cn2ncc(C)c2)=O)CCN(C(=O)CC2CC(C)(C)C2)C12CCC2 CC(C)C(C(=O)N1CCC(OCNC(=O)CO)CC1)SCc1ccccn1 N1(C(c2nccc(C#C)c2)=O)CCC(NC(=O)C(C)(C)SC)C(C)(C)C1 n1(CC(N)=O)cc(COCC(N2CCC(CNC(N)=O)C2)=O)nn1 CCC(C(=O)NC(C)CCNC(=O)Cc1ncc(Cl)s1)C(F)(F)F c1(OCC)ccccc1CC(=O)NC1(C(N(C)CC2(COC)CC2(F)F)=O)CC1 N1(C(CCOC)=O)CCC(NC(=O)C=C2CCCCC2)C(CO)C1 N1(C(CCCC=C)=O)CC2(COC)CC1(C(=O)NCC1(CCO)CCCC1)C2 c1(C2CC(SCC3CCCN3)C2)cnc(NC(=O)OC(C)(C)C)cn1 C(=O)(C#CC1(C)CCCO1)NCc1ccc(C(N2CCC(C#C)CC2)=O)s1 C1(C(=O)NCCn2cc(CNC(C(C#C)(C)C)=O)nn2)CCC12CCCO2 C12(NC(C(C(C)NC(=O)COC3CC=CC3)(C)C)=O)CCCN(CCC1)C2 C1(C(C)C)C(NC(=O)CCC#N)CCN1C(C1CC1C#N)=O CC(C)(C)C(C(=O)NCCOCCCNC(=O)Cn1ccnn1)C1CCCCC1 C1(C(N2CC(NC(C3(F)CCCC3)=O)C2)=O)(CC)CCOC1 c1(C(N(C)CCOCCC(=O)NCC2(C)CCC(=O)N2C)=O)cccc(C)c1F C1(CC(=O)NC(c2cncn2C2CC2)C)C2CN(C(=O)C(C)c3ccco3)CC12 n1(C(C)C)nccc1C(N1CCCC1CNC(C1(C)CC1)=O)=O CCCC(CCCNC(=O)C(C(F)(F)F)OC)NC(=O)C(=O)NC12CC(C1)C2 C1(CC(=O)NCc2cn(CC)nn2)CC2(CC2)CN1C(c1ccc(OC)nc1)=O CN1CC(O)CC1(C)C(=O)Nc1ccc(-c2cncc(F)c2)c(F)c1 CCCCCCCCNC(=O)C(=O)NC1CCC(NC(C2C(F)(F)C23CC3)=O)CC1 C1(C(C)C)CN(C(c2cc(C3CC3)on2)=O)CCN1C(c1cn2ccsc2n1)=O C1(C)(C(N(CCNC(c2cccc(OCC)c2)=O)C2CC2)=O)CCCNS1(=O)=O c1(CC(N2CC(O)(CCc3cn(CCO)nn3)C2)=O)c(F)cccc1Cl.C(=O)OC CCC(CNC(c1ccc(C2CC2(Cl)Cl)cc1)=O)(CC)NC(C1CC1C)=O c1(C(=O)NC2CC(C)N(C(=O)CC(=O)N(C)C)CC2)cccc2c1CCC2 C1(NC(C(C)OCCOCC)=O)CCC(CC(=O)NC2CSC2)C1 C(=O)(C(C(C)C)c1cnn(C)c1)N1CC(C)(NC(COCC(C)C)=O)C1 C1(NC(C(n2c(C)cc(C)n2)C)=O)CC2CCC1N2C(C1CC12CCSCC2)=O c1(NC(C(CNC(C(C)SCCCC)=O)CC2CC2)=O)cccc(C)c1O C1(C(C)COC)CCN(C(c2cnc(O)n2C)=O)C1C(N1CC(N2CCNC2=O)C1)=O C(CCC(=O)N(C)CC=CC(N1CCC(Cc2nn[nH]n2)C1)=O)=C(C)C C1(F)(C(=O)NC(c2ccccc2)CC)CCN(C(C2(C)CCC3CC3C2)=O)CC1 C(=O)(CCCCN=[N+]=[N-])N1CC(C)(C)C(C(N2CCCCCCC2)=O)C1 N1(CC(=O)OC)CCC2(CC1)CC2(C)C(N1CCCC(C)C1CN)=O C=C(C)CC(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(=O)Cc1ccc(O)cn1 c1(NC(C2C3(CCN(Cc4ccc(OC)nc4Br)C3)C2)=O)c(F)cc(Br)cc1Br N1(C(N)=O)CCCCC1C(=O)NCC(=O)Nn1cc(C(C2CCOC2)O)nn1 N1(C(C(=Cc2cccnc2)C)=O)CCCCC(NC(c2ccc(Cl)cc2Cl)=O)C1 C=C(C)C(C)(O)C(=O)NCC(C)(CO)NC(c1ccc(COC)o1)=O c1(NC(=O)Nc2ccc(C(F)F)nc2)nc2ccccc2n1CCOCCO c1(C(c2nnnn2C)Nc2ccnc(OCC)c2F)cc(C)cc2c1CCC2 C1(C(=O)NC2(C(=O)NC)CC2)CC2(CCC2)CN1C(=O)C(C)(F)C(=O)OC N1(C(CC(=O)OCC)=O)CC2CN(C(=O)C(C)Oc3ccccc3)CC2C1 n1(CC2CC(C)C2)nc(-c2cccc(Br)n2)nc1-c1cn(C(F)F)cn1 c1(C(=O)NCCC2(CNC(C(C)C#N)=O)CC2)cc(O)nc(O)n1 C(=O)(CCS(=O)(=O)C1CCCC1)NCC1(C)CCN(C(C2CCC(=O)O2)=O)C1 c1(C(=O)NC2CCCCN(C(C(C)(C)CC3CC3)=O)C2)ccc([N+](=O)[O-])cn1 C(=O)(C(C)(C)CCF)NCCCNC(c1ccnn1CC1CCC1)=O.CN1CC1 CCC(CC(=O)N(C)Cc1ccc(N2CCC(C)C2)nc1)OC C1(C(N2CC3(N(C(CC(C(C)C)C)=O)CC3)C2)=O)CCC2(CC1)CC2(F)F N1(C(c2nc(C(C)=O)sc2)=O)CCOCC1CNC(c1ccnc(C(N)=O)c1)=O c1(CCC(=O)NCCOCCN(C(C(=O)NC)=O)C)nccn1C.C1C(=O)N1 Cc1cc2cc(NC(=O)N(CCCF)C)ccc2cn1 C(=O)(CCCCC(=O)NCC(=O)NCc1ccc(Br)c(F)n1)NC CC(CCCc1ccccc1)C(=O)NCC1CC1NC(c1ccc(CC2CC2)s1)=O S(=O)(=O)(CC(=O)N1CC2CC2(CNC(=O)CCC2CCCCC2)C1)N(C)C Cc1ccc(C(=O)NCC(C2CCCN2C(C2CCC(C)CC2)=O)(C)C)cc1C C1(CC(N2CC3CCN(C(CCC)=O)CC32)=O)CCc2sccc2C1=O N1(C(c2cc(C(=O)OCC)n(C)n2)=O)CCC(NC(c2coc(Cl)n2)=O)C(C)C1 N1(S(C(C)C)(=O)=O)CCC2(CC1)CC2C(N1CCCCCCC1C)=O n1(CCC)ncc(C(=O)NC(C)(CNC(C2CCCCC2CC)=O)C(C)C)c1C N1(C(c2cc(CNC(C3N(C)CCC3)=O)oc2)=O)Cc2n[nH]cc2C1CO C1(NC(C2C3(CC(C)(C)C3)C2)=O)CCC2(CC1)CN(C(C1CCCC1)=O)C2 c1(C(=O)NCCC(C)NC(c2nc[nH]c3nccc2-3)=O)ccnc2[nH]c(O)nc12 C=CCC(CNC(c1cc2occc2[nH]1)=O)C(=O)NCCCOC(C)C c1(N2CC(F)(C(=O)NC(c3ccccc3)CO)C2)ncc2[nH]cc(I)c2n1 c1(C(N(C2CCC(NC(C(C)n3cnnn3)=O)CC2)C)=O)ccc(O)c(N)c1 C1(NC(Cn2c(C)nnn2)=O)CCCCC1CNC(=O)CNc1nccs1 C(=O)(C(C1=NOCC1)N1CCC(C(O)C(F)(F)F)CC1)NCC1(C(N)=O)CCC1 c1(N(CC(C)C)C(=O)OC(C)(C)C)nc2c(c(=NCCOCCCO)[nH]1)COC2 C1(OC)CC(F)CN(C(=O)C2=CCC(NC(=O)CCC(C)SC)C2)C1 c1(OC)cnc(C(=O)N(C2CCC(NC(c3nnc(C(C)(C)C)s3)=O)C2)C)cn1 Cc1cc(C#N)ccc1C(=O)NCC1(CN(C(=O)CC2CN(C)C2)C)CC1 C1(C(=O)OCC(CC)NCCC2CC2)CC2CCC1CC2 Cc1cc(C(=O)NC2CCC(CC(=O)N(C)CC3CCCO3)CC2)ccc1C#N Cc1ccc(C(=O)N(CCCCC(=O)NOCC2CC2)C2CC2)cc1C#N Cc1cc(C(=O)NC2CCC(NC(C3(C)CC(C)C3)=O)CC2)ncc1N N1(C(CC2N(CC)CCC2)=O)C2CCC1CC(NC(C1CN(C(C)C)C1)=O)C2 c1(C(C(=O)NCC(C)C)N(C2CC2)CC2(C)CCC2)ccc(Br)cc1F N1(C(c2c(C(C)(C)C)ncs2)=O)CCCC(C2CCNC2)C1 Cc1c(F)ccc2[nH]c(C(N3CC(C(C)(C)O)(CNC(=O)CN(C)C)C3)=O)cc12 c1(C(=O)NC2C(C)CCC2)cccc([N+](=O)[O-])c1Br C1(NC(CC2N(C)CCC2)=O)CCCC(C(N2CCC(O)(C(F)F)C2)=O)C1 CC1CC=CCC1NC(C1(CO)CCN(C(c2cccc[n+]2[O-])=O)C1)=O C1(CNC(CC(=O)NC)=O)CCCC12CN(C(c1c(C)cc(Br)cc1Cl)=O)C2 c1(C(=O)N=c2cccn[nH]2)ccc2[nH]cc(C3=Cc4ccccc4C3)c2c1 c1(CNS(CC(C)C)(=O)=O)cc2ncccc2o1.N12CC3(CC1CO3)C2 c1(CC)cccc(C(c2nnnn2CC2CCC2)NCC(N)=O)c1 Cc1cc(F)c(CNC2CC(NC(C3CCSCC3)=O)C2)cc1Br CC1C(NC(C2CCC(=O)NC2)=O)CCCN1C(=O)CC(c1ccc(O)cc1)=O C(=O)(C(C)SCC)N1CCC1.C(=O)(CN(CCCF)C)NC(=O)NCC c1(NC(C2(NC(=O)CCCn3ccnn3)C(C)(C)C2)=O)ccc2nccn2c1 Cc1cnc2c(C(N3CC(C)(NC(C4CCCC(C)(C)O4)=O)C3)=O)cccc2n1 N1(C(C2(C#N)CC2)=O)CCN(C(c2ccc(C(C)C)c(Br)c2)=O)C2CC12 c1(COC)nc(C)c(C(=O)NCCC2CC(NC(c3c[nH]c(Br)c3)=O)C2)s1 CCCCC(F)C(=O)N(C(C)CC(=O)NC1CCOC(C)(C)C1)C C=CCCC(C(=O)NCCn1ccnn1)NC(c1coc(SC)c1)=O CC1CCCC(C)CN1C(=O)CC(C(F)(F)F)c1ccon1 c1(C(C)C(=O)NC(CNC(=O)Cc2nccn2C)C2CC2)ccc(Cl)cc1 C1(NC(=O)CCC2CCCCO2)C2CN(C(=O)CC3CC(F)(F)C3)CC12 CC(CCNC(c1n[nH]cc1F)=O)CCNC(c1cc(-c2ccccc2)on1)=O C=CC(C)(O)C(=O)NC(C1CCN(C(=O)CCCOc2ccccc2)C1)C CC1(C)C(NC(c2n[nH]c(=N)[nH]2)=O)CC1C(N1CC(n2cccn2)C1)=O C1(C)(CNC(c2c(CC)n(C)nc2)=O)CN(C(c2nc(Cl)oc2C)=O)CC1C C1(CC(=O)NC(CNC(C(C)NC(C)=O)=O)(C)C2CCC2)CCCC(C)(C)O1 N1(C(c2ccc(CCC)[nH]2)=O)CCC2(CNC(=O)CCC[N+](=O)[O-])CCCCC12 C(=O)(C(CC(C)(C)C)OC)N1CC(C(N2C(CC(=O)NC)CC2)=O)OCC1 c1(C(=O)NC2(CO)CCN(C(CNC(CC)=O)=O)C2)cc2c(C)cccc2o1 c1(OC(CCNc2ccc(S(C)=O)cc2)=O)nc2ccc([N+](=O)[O-])cc2s1 c1(C(N(CCF)CC)=O)ccc2c(n1)CN(C(C1CCC(C)(C)CC1)=O)CC2 CC(C(C)(C)C(=O)NCc1ccccc1)NC(=O)CN(C)C N1(C(C(C)NS(CCC)(=O)=O)=O)CCC(C2CCN(C(=O)CC(=O)OC)CC2)CC1 c1(C(N2CC(CCNC(=O)C(F)C3CCOC3)OCC2)=O)ccc(CO)c(Cl)c1 CCC(CC(=O)N1CC(OC)CC1CCNC(=O)COCC(F)F)OC c1(CC)ccc(CCOc2ccc(NC(N3CCN(CC)CC3)=O)cc2)c(C)c1 C1(O)(C(=O)NCCCCCN(C(C=NOC)=O)C)CCCC(C)(C)C1 C=CCC(C(=O)NCC#CC(=O)N1CCC(CCCC)C1)OC c1(C(N2CC3N(C(c4cn(C(C)(C)C)nc4)=O)C3C2)=O)cc(O)cc(Cl)c1 C1(C(c2n(C3(C)CC3)nnn2)NCC2CC(c3ccccc3)C2)CCCCC1C c1(C(=O)NCC(C)(C)O)ccc2c(n1)CN(C(=O)CCCS(C)(=O)=O)CC2 C1(NC(COCC=C)=O)CCCC(n2cc(C3(C)CC3)nn2)C1 Cc1ccccc1N(C(=O)CCN(CCO)C(c1csc(F)c1)=O)C CN1CC=C(CC(=O)N2CC(CNC(=O)CSCc3ccccn3)(OC)C2)CC1 C1(CNC(c2c(C)cns2)=O)CN(C(=O)C=Cc2ccncc2)CCCO1 N1(C(C(CNC(C(C(C)C)NC(C)=O)=O)C(C)C)=O)CCCC2(CC1)CC2 c1(C(=O)NCC(C)N(C(C2=CC(C)(CC)C2)=O)C)cc(Cl)cc2c1CCC2 c1(C(C(=O)NCC(C)C)N(C)CC2CC2(C)C)ccc2ccn(C)c2c1 N1(CC(N2CC3C(CNC(c4c(C)nncc4)=O)(C3)C2)=O)CCc2ccccc21 c1(C2(CO)CCC2)ccc(OC(F)(F)F)c(Cl)c1.C12CN(C1)C2 C1(=CC(=O)NCC(C(=O)NCC(C#C)CC2CC2)N(C)C)CCC(C)CC1 C(=O)(CC(C(N)=O)c1ccccc1)N1CC(C)C1.C(C(C)C)(c1nnnn1C)N C1(C)(C(=O)NCC(C)NC(=O)CNC(=O)C(C)(C)C)CCCC1C C1(O)(CC(=O)NC2CC(O)(CNC(=O)C(F)CC3CCCCC3)C2)CCCC1 Cc1nscc1NC(=O)N(C(C)(C)CCN1CCCC1)C1C2CCCC12 C1(NC(C2(OCC)CC2)=O)CCN(C(=O)COC2CC2)CCC1COC Cn1cnc(NC(=O)CC2(C)CC2(Cl)Cl)n1 N1(C(CC2(C=C)CCC2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 c1(C(=O)OCC)cccc(Nc2cc(C(F)(F)F)nc(C)n2)c1C N1(C(c2cccnc2Cl)=O)CC(C2CCN(C(C3(C(F)F)CC(O)C3)=O)CC2)C1 N1(C(C(COC)(F)F)=O)CCc2nc(O)cc(C(=O)NCC3(C)CCCO3)c2C1 C1(C(=O)OCC=CC2CC2)CC(C2CCOCC2)=NO1 C1(C(=O)OC)C(C(=O)NC(CC(C)=O)C(=O)OC)C12CC2(F)F N1(C(C2(F)CCN(C(c3c(C)n[nH]c3C)=O)C2)=O)Cc2c(O)n[nH]c2C(F)(F)C1 CN1CCCC(C(N2CCC(CC(=O)N(C3(c4cc[nH]n4)CC3)C)C2)=O)C1 C1(C(N2CC(CC(C(=O)NC(c3cn(CC)nc3)C)F)C2)=O)CC(=O)CCO1 C1(NC(CC(C)C)=O)COC2(CCN(C(c3cccnc3S)=O)C2)C1 C1(C(=O)Nc2cn(CC#C)nc2)(CC=C)CCN(C(C2(C)CCNC2=O)=O)C1 C(=O)(C(C(C1CC1)OC)N1CCC(OCCC#N)CC1)NCCCC C1(CN(C(Cc2cc(C)[nH]n2)=O)C)CCCC(NC(C2(C)CCCC2)=O)C1 N1(C(C(CC)CC)=O)CC(C(=O)NCCC2CCCC(C)C2)C(C)(C)C1 C(=O)(C(CNC(c1cnnc(O)c1)=O)CC1CC1)NCC(C)CC1CCCC1 c1(C(N2CCCC2CNC(C2(CO)CCCC2)=O)=O)csc(-c2cnc[nH]2)n1 C1(C(=O)NCCN(CCC)C(c2sccc2OC(F)F)=O)CC2CC1CO2 N1(c2n(C)c(Cc3ccc(Cl)cc3F)nn2)CCc2nc[nH]c2C12CCNC2 C1(C)(COC)CCCN1C(C1CN(C(=O)C(c2cnn(C)c2)C)C1)=O c1(C(N2C(CN(c3ccc(OC)nc3)C)CCC2)=O)cc2n(n1)C(C)CCC2 c1(CNC(C2C(C)(C)C2)=O)nccn1O C(=O)(CCCCCOCC)N1CCC(CNC(C(C(=O)OCC)C2CC2)=O)C1 c1(CNC(C2CC2C(=O)NC2(c3ccccc3)CC2)=O)ccc(Cl)cc1Cl C1(NC(C(c2cccc(F)c2)C)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC1C N1(C(C(CCSC)NC(=O)CCc2cccnc2)=O)CCC(F)(F)CC1C N1(C(C(C)C2CCOC2)=O)CC(C)(C)CC1CCC(=O)NCCOC1CCCC1 N1(C(C(CC=CC)CC)=O)CC2CCN(C(=O)Cn3ncn(C)c3=O)CC(C2)C1 C(=O)(C(F)(F)C(O)C1CC1)NCC1(NC(C(C)n2cccn2)=O)CCCC1 c1(C(N2CC(NC(c3c(OC)n[nH]c3)=O)C(CO)CC2)=O)cccc2ncsc12 c1(C(N2C(C)(CNC(CC(C)OC)=O)CCC2)=O)cc(C)nc(Cl)c1 C1(C(=O)NC2CC(CCNC(C(C)Sc3ccccc3)=O)C2)CC2CC2CC1C C(=O)(C1=CCC(C)CC1)N1CCC(C)(CC(=O)NCC(CSC)OC)C1 c1(CC(=O)NCC(c2ccc(F)cc2F)C(=O)O)c[nH]c2cccc(Cl)c12 c1(CC)cc(C(=O)NOCC(=O)N(CCS(=O)CC)CC(C)C)no1 Cc1cc(C(=O)NCC(=O)NC(C)CCCNC(=O)Cc2nc(C)cs2)cc(C)c1 N1(C(c2ccc(C#C)cc2F)=O)CC2CCN(C(=O)CCC3CCOC3)CC2C1 N1(C(C(CC=C)CNC(c2cc(Cl)ns2)=O)=O)CC2CC(C1)C2(C)C c1(NC(=O)Nc2nnc(CC3CC3)s2)cccc(Cn2cc(Br)cn2)c1 c1(C(C(=O)OC)OC(=O)C(c2ccccc2)OC)cc(C(F)(F)F)cc(Cl)c1 C#CCCC(=O)NCCC(C)NC(c1cn(Cc2nc(C)cs2)nn1)=O CC(C)(C)CC(O)C(=O)NC1CN(C(=O)CCc2ccc(Cl)s2)CC12CC2 C(=O)(CC1COc2cc(O)ccc21)NCCC(C)NC(=O)C#CC1CCOCC1 C(CC(C)C)(C(N)=O)N(C(=O)OC)C.N12CCN(CC1)C(C(F)F)CNC2=O c1(C(=O)NC(C(CO)NC(c2c(CC)sc(=N)[nH]2)=O)C)nnc(C)cc1O CCCCCS(=O)(=O)N(C(C)(C)CCC)C C1(C)(C(=O)NC(C2CN(C(C(CC=C)NC(C)=O)=O)C2)C)CCC(F)(F)C1 O=C(C1CC=Cc2ccccc21)NC1CCC(NC(C2CCCC2)=O)CC1 c1(C(N2CCCCC2C2CC2)C(=O)NCCOCC)ccc2c(n1)CCC2 c1(C(N2CC3CN(C(c4ccc(Br)c(Cl)c4)=O)CC32)=O)cc(F)c(F)c(Br)c1F c1(C(N2CCC(C(C(N3CC(CCCCC)C3)=O)C)CC2)=O)cc(C)nc(O)n1 C1(C(N2CC(O)(CCNC(c3c(C)nns3)=O)C2)=O)CCC(=O)N1C C1(C#N)(C(=O)NC2CCCC(CNC(c3cc(OC)n[nH]3)=O)C2)CC2CCC1C2 N1(C(c2c(C)cns2)=O)CC(CNC(=O)CC2C(C)(C)C2(C)C)OC(C)(C)C1 c1(C(=O)NCCC2(NC(C3CC4C=CC3C4)=O)CCC2)ccc(F)cc1F c1(C(=O)NCC2CN(C(COCCC)=O)CC2O)cnc2ccccc2n1 c1(-c2cn(C3CCC(C(=O)NCCCN(S(C)(=O)=O)C)C3)nn2)ncccc1F C(=O)(CP(=O)(C(C)C)C(C)C)N(C(CNC(c1ccc(C)c(N)c1)=O)C1CC1)C C1(C(=O)NCC2C(CNC(CSC)=O)C2(F)F)OC(C)(C)OC1(C)C c1(CC(=O)NC(CNC(C2CC(C(C)C)C2)=O)C(C)(C)C)cn2c(n1)CCCC2 c1(C(=O)NC2CCN(C(c3cnc(CC)[nH]3)=O)C2C)ccc(F)c(F)c1F N1(C(C2C(C)OCC2)=O)CCN(C2CN(C(C3(C(F)(F)F)CC(O)C3)=O)C2)CC1 C(=O)(C1=CC2CC(C1)CC2O)NCCCCC(CO)NC(c1n(C)ccc1)=O Cc1cc(NC(C2CCN2C(c2nc(Br)cs2)=O)=O)cc(Cl)n1 c1(NC2C(NC(CC(CCC)O)=O)CS(=O)(=O)C2)nc(Cl)nc2c1cnn2C(C)C C=CCCCCCC(=O)NCCCC(C)(C)NC(c1cc(C)cnc1C)=O Cc1cnc(C(=O)NC2CCC(NC(c3cn(CCCF)nn3)=O)CC2)cc1C c1(NC2CCN(C(CCCCCOCC)=O)CC2C)nc(C)nc(O)c1C C(=O)(CC1CCc2ccccc21)NC1C(CNC(C2CC(SC)C2)=O)CC1 Cc1c(CO)cc(C(N2CCCC(CNC(C3(CNC(N)=O)CC3)=O)C2)=O)n1C N1(c2c(C)c(N(C)Cc3ccccc3Cl)ncn2)CCC2(CC1)CCC2(C)C c1(C(CO)NC(=O)NC(C(C)C)CC2CCNCC2)ccc(F)cc1F C1(CCNC(C(n2ncc(C)c2)C)=O)CSCCN1C(c1ccoc1)=O c1(OCCCCC)ccc(C(=O)NC(C)CNC(=O)C=Cc2csc(C)n2)cc1 N(C1c2ccccc2CC12CCCC2)C(=O)NC(C)(C)C.Cc1cccc2c1CCC2 Cc1ccc(O)c(CC(=O)NC2CN(C(C3C4CCCOC34)=O)CC2CO)c1 CC(C)(C)CC(O)C(=O)NC1CC(F)(CNC(=O)CCCC(N)=O)C1 N1(C(C(C)C(F)(F)F)=O)CCN(C(=O)C(=O)N(C)C)CC12CC2 N1(C(c2cnn(CC)c2C)=O)CCN(C(c2ncc3ccccn23)=O)C(C)C1C C1(NC(CSC)=O)CC(C)N(C(C2(SC)CCC2)=O)C1 C1(C(NOCCOC)=O)C2CCN(C(=O)CC3CCC(C)C3)CC12 C1(C(=O)NC(CN(C)C(c2cnc(O)s2)=O)(CO)CO)CC2(C1)CC(F)(F)C2 C1(N(CCCn2nccn2)Cc2ccc(Cl)o2)CC2CC1CN2 Cc1nccc(C(=O)NCC(CC2CC2)C(=O)NCCC2CCCC(C)C2)n1 C=C(C)CCN=c1[nH]c2c(c(=NCCCCN3CCCC3)[nH]1)COCC2 N1(C(C2=CCC(C)CC2)=O)CCCC2(CCCCC2NC(c2cnn(C)n2)=O)C1 C1(CNC(CC(C)NC(N)=O)=O)CCN(C(C2CC3(C2)CC(F)C3)=O)CC1O CC(C)C(O)C(C)C(=O)NC1(C(=O)NCC2CCCCS2)CCCCC1 c1(C(CCOc2ccc(Br)cc2)Cc2n(CC)cnn2)cccc(C#N)c1 C1(NC(C(c2cc(F)cc(F)c2)(C)C)=O)CCCCN(C(C2CCCCO2)=O)C1 N1(C(C2(N(C)C)CCC2)=O)CC2C(C(F)(F)F)CC2(NC(=O)CC2(C)CC2)C1 CCCC(C)(CC)C(=O)N(C(C)CCNC(c1cncs1)=O)C c1(C(=O)NC(CC)C2CCC2)cc(=NC(=O)C=Cc2ccc(C)o2)[nH]n1C c1(NC(C2CCCN(C(Cc3c(C)nn(C)c3)=O)C2)C)ncnc2cc(Br)sc12 C(C(C(=O)N1CC2CCC1CC2NC(=O)C(C)(F)F)C(F)(F)F)OC C=CC1CCCN1C(=O)C(C1(O)CCCCC1)NC(=O)CSC(C)C CN1Cc2ccc(C(N3CCN(C(c4ccon4)=O)C4CC34)=O)cc2C1 c1(CC)cc(C(=O)NC(C)C(C)NC(c2ccccc2CO)=O)cc(C)c1 C=CCC(CNC(C1CC(C)=NO1)=O)C(=O)NCCC(C)(C)F c1(C(=O)N(C2CCNC2)CCc2ccn3nccc3n2)[nH]c2ccccc2c1Cl C1(C(N(C(C)CNC(=O)CCc2cn(C)nn2)C)=O)Cc2ccccc2N1C Cc1cc(C)cc(C=CC(=O)N(CC(C)NC(=O)C=CC2CCOCC2)C)c1 N1(C(c2ccnc(C3CCC3)c2)=O)CC2(C1)CN(C(C1(CC=C)CCC1)=O)C2 C1(NC(CNC(CC)=O)=O)CC2CCCC(C1)N2C(=O)CC1CCCCO1 CCCC(C(=O)NC1(CO)CN(C(c2ccc(Cl)c(CC)c2)=O)C1)C(C)C C(=O)(C1c2ccnn2CCN1C(=O)OC(C)(C)C)NCCc1cc(C)c(F)c(C)c1 c1(CC)cc(C(N2CCC(NC(c3ccc(F)cn3)=O)C2)=O)cc(N)c1 c1(CN(C(CNC(CC2(OC)CCC2)=O)C)C)ccc(C)nc1F CC1(NC(=O)C=CC2CCCO2)CC(NC(C2CCCSC2)=O)C1 c1(C(=O)NCCC2CCCN2C(=O)C=CC2CC2)cccc(F)c1O N1(C(c2ccc(CC(C)C)o2)=O)CC(NC(C2(C(F)(F)F)CC2)=O)C(C2CC2)C1 C12(NC(=O)CCOCc3ccccc3)CC(C1)N(C(=O)COCC(F)F)C2 NC(=O)N=Nc1ccc(C(=O)NCc2[nH]ccc(=O)c2O)cc1 N1(C(=O)CSC2CCCCO2)CC2CCC1CN2C(C1(C2CC2)CCCO1)=O Cc1nc2cc(C(N3CC(CO)CCC3C)=O)ccc2n1C1CCOC1 Cc1cc(CNC(C2(C)CCCN2C(=O)C(C)Cc2ccccn2)=O)cc(C)c1 C=C1CC(NC(=O)NCC2CCSC2)C1 C1(C)(CC)C=C(C(=O)NC2CC(C(C)NC(c3cnccc3C)=O)C2)C1 n1(CC(=O)NC(C2CCC(NC(=O)Cc3ccsc3Br)C2)C)nnc(=N)[nH]1 c1(OC)cc(CC(=O)N(C)CCNC(=O)C2CC2)ccc1C c1(C(=O)NC2C3CN(C(CC(=C=C)C)=O)C2C3)cc2cc(Cl)cnc2[nH]1 c1(C(N2CC3CCC(C2)N3C(c2ccc(CO)o2)=O)=O)nncc2ccccc12 Cc1ccc(CNC2CC(NC(c3cnc(O)s3)=O)C2)c(Cl)n1 C12(CNC(C(c3ccco3)NC(C(C)=C3CCCC3)=O)=O)CCCN(CC1)C2 C(=O)(C1COc2ccc(Br)cc21)N(CC(C)(C)CNC(=O)CSC(C)C)CC C1(NC(c2ccc(Cl)c(Cl)c2)=O)CC2(C1)CC(NCc1cc(Cl)cnc1F)C2 c1(C(N2C(CN(C)C(C3CCC(=O)C3)=O)CCC2)=O)ccc2nsnc2c1 N1(C(C(c2cccc(Br)n2)C)=O)CCN(C(C2(O)CCC2)=O)CC1CF Cc1cc(N2CCCC(c3nc[nH]n3)C2)nc(NC(c2nccc(O)n2)(C)C)n1 C1(CNC(C(C)OCC#C)=O)CC2(CO1)CN(C(=O)C(C)=C1CCCC1)C2 CC1(C(=O)NCC(CC(F)(F)F)NC(=O)CNS(C)(=O)=O)CCCCC1(F)F c1(C(N(C2CN(C(CCCCCOC)=O)C2)C)=O)cc2c(cn1)CCCC2 Cc1cccc(CC(=O)NC2CS(=O)(=O)CC2NC(c2cccc(=O)o2)=O)c1F c1(C(=O)OC)cc(OC)ccc1NCCO.N12CCCC(C1)OCC2 c1(C(=O)NCC(CCCC)NC(=O)CNC(=O)C(C)CC)cc(O)ccc1Cl CC1(C(=O)NC2CCCCC2NC(c2ccc(F)s2)=O)CCC(=O)N1 N1(C(C)=O)CCCN(C(C2(CF)CCN(C(=O)C3CC3)C2)=O)CC1 Cc1ncc(C(=O)NCC2(C)CC(NC(=O)CSCC(F)F)C2)cn1 C(=O)(C(F)CC(C)(C)C)N1C(C)CCC(C(=O)NCc2c(C)nsc2)C1 C1(CNC(c2c(CC)nc[nH]2)=O)CC(C(C)(C)C)CCN1C(=O)CC(C)OC c1(C(C)N(Cc2ccccc2N2CCCC2)CC)ccccc1C(F)(F)F C1(NC(=O)CC23CCCC2C3)CCCCC12CCCC2 c1(C(N2CCC(OC)CC2C)C(=O)Nc2c(OC)cccc2)cnccc1C#N N1(C(CCS(C)(=O)=O)=O)CCC(C2CCCN(C(=O)C3=C(Cl)CCOC3)C2)C1 C1(C)(NCCC(C)NC2COC2)CCCCC1O C(CCC(C(=O)N1CCCC(C(C)O)C1)NC(=O)C(C)C(F)(F)F)OC N1(C(CC2N(C)CCOC2)=O)CCC(NC(=O)CCc2nc(O)n[nH]2)C(F)C1 C1(C2(O)CN(C(C3CC(=O)N(O)C3)=O)C2)(CNC(CC2(OC)CC2)=O)CC1 N1(c2c(C(=O)OC)cccn2)CCC(NC(=O)CCCNC(N)=O)C(CO)CC1 c1(C(N2CCC(C)(NC(C(C)CC(N)=O)=O)C2)=O)cn2cc[nH]c(=O)c2n1 CC(C)CC(=O)NNC(=O)Cc1nc(Cc2ccccc2)ns1 N(C(=NCCC(C)N1CCOCC1)NC(C)COC(F)F)C(c1ccccc1)C#C C(CCC(C(=O)N=c1ccn(C(C)C)[nH]1)NC(=O)C#CC(C)C)OC C(=O)(C(C)CC(=O)N1CCN(C(c2ccc(F)nc2)=O)C(C)C1)OC c1(C(=O)NC(CN(C)C(C2CCC(C)(C)CC2)=O)(C)C)ccc2c(c1)OCCN2 Cc1cc(C(=O)N(C)CCN(C(=O)CC2CCCC23CC3)C)sc1C CC1CN(C(c2ccoc2)=O)CCN1C(c1cn(CC2CNC(=O)O2)nn1)=O N1(C(=O)CO)CC2COCC2(C(N2CCN(c3ccccc3)CC2)=O)C1 c1(C(=O)NCC2CC(NC(c3cn(C)nc3)=O)C2)ncn2c1CCC2 C(N=c1[nH]cc2ncnc-2[nH]1)C1(C)CCN(C(c2cc(COC)oc2C)=O)C1 c1(OC)cccc2ncnc(N(C(C)CCNC(C3CCOC(C)(C)C3)=O)C)c12 c1(C(=O)NC2C(NC(=O)CC3CC=CCC3)CC2)ccc(F)c2cccnc12 c1(NCCC2CCCN(C(C3C(OC)CCC3)=O)C2)ncnc2c1CCC2 C1(NC(C2(NC(C3CC4COCC4C3)=O)CCN(C)C2)=O)CCn2ncnc2C1 C(C)(c1ccccc1)=CC(=O)NCc1cn(CCNC(C(CC2CC2)OC)=O)nn1 C#Cc1cnc(C(=O)NC2CCC2C(=O)NC2CCC(CN(C)C)CC2)c(C)c1 c1(OC)nc2c(s1)CCCC2.N1C(=S)NC2CC2C(OC)C1 C12(C(=O)NCC(CNC(=O)Cc3ccccc3)F)CCC(O)C1CC2 C1(C(N2CC(CCCCNC(C(C)OC)=O)C2)=O)C2CC1(c1ccccc1)CO2 c1(C(C)C)nc(C(=O)NC(C)CN(C(=O)C(C)Cc2ccccn2)C)co1 CCCCC(C)C(=O)NCC(C)(F)CNC(c1ccnc(N(C)C)c1)=O C1(C(N2CCN(CCOC)CC2)=O)CC(F)CCN1C(=O)CCC(C)(C)C c1(CC)[nH]nc(C(N2CCC(CCNC(c3cocc3C)=O)CC2)=O)c1Cl CC1C(NC(c2ccnc(F)c2Cl)=O)CCCN1C(=O)C(c1ccccc1)F c1(CC(=O)NC2C(NC(=O)CCc3cnc[nH]3)C2)ccc(Cl)c(F)c1 C(=O)(C(C)(C)CC(F)(F)F)N1CCCC(c2cn(C(CCCCCC)CC)nn2)C1 N1(C(C2CCS(=O)CC2)=O)CC(C2CN(C(C3CC4(C3)CC43CC3)=O)C2)C1 S(=O)(=O)(CCC(=O)N(CCC(C)NC(c1ccc(C(O)CF)cc1)=O)CC)NC Cc1cccc(CNC(=O)C(c2cn(C)nn2)NC(c2ccnnc2C)=O)n1 c1(C(=O)NCC2CN(C(CCc3c(NC)cccc3)=O)C2)ccnc(C)c1O c1(C(N(CCN(C(C(C2CCCO2)OC)=O)C(C)C)C)=O)ncn(C(C)C)n1 C(C)(CC)(CCNC(=O)COc1cnn(C)c1)NC(c1ccn(CCC)n1)=O C1(NC(CC(C(=O)OC)C)=O)CC2CCC(C1)N2C(=O)CSc1ccncc1 C1(NC(=O)CN(C2CCC2)C(C2CCS2(=O)=O)=O)CCOCC1F N1(C(C(C2CCN(C(c3cnc(C)nc3)=O)CC2)C)=O)CCC(CO)C(C)C1 C#Cc1cnc(C(N2C(C(=O)N(CC#CC)CC)CCC2C(C)C)=O)c(C)c1 c1(C(=O)NC2C(CO)CCN(C(CCC(CC)C)=O)C2)cnc2c(ccn2C)c1 C(=O)(C(F)(F)CO)NCCC1CC(NC(C2(C(=O)NC)CCC2)=O)C1 C1(NC(C(C)(C)OC(C)C)=O)CC1C1CCCN(C(=O)C=CBr)C1 N1(C(C(C)N=[N+]=[N-])=O)CCCCC2(CCN(C(C3Cc4nccn4C3)=O)C2)C1 c1(CN(C(=O)C(=C2CCCCC2)F)CCO)cc(Br)c(F)c(F)c1F Cc1nn(C)cc1C1=NOC(C(N2CCCC(NC(c3ncn(C)n3)=O)C2)=O)C1 C(N=c1ccnc(NC)[nH]1)C1N(CC2C(CC)CCC2)CC1.C12CC(=O)N(C1)C2 CCC(CC(C)C)C(=O)N(CCCNC(=O)C(C)n1ccnn1)C(C)C C(CCCC1C(=O)N1)(OC)OC.c1(CC(C)NC(=O)C(C)(C)C)ccc(F)cc1 c1(C(=O)NCC2CC3CC3N2C(=O)C(O)C2CC2)cc(Cl)ccn1 C=CC1CCN(C(C2N(Cc3c[nH]nc3-c3ccc(C)cc3)CC2(C)C)=O)CC1 c1(CN(C)C(c2cccc(O)c2)=O)ccccc1CN1CCC(O)C1 CCC(C)(CC)C(=O)NC1CCOCC1C(=O)NC1CC(n2cncn2)C1 N1(C(C2CN(C)C(=O)C2)=O)CCCC2(CCN(C(c3ccn(C4CC4)n3)=O)C2)C1 Nc1cc(C(=O)NC2(CO)CN(C(C3CC(=O)NC(=O)C3)=O)C2)ncc1F C1(C)(CC)NC(=O)N(CC(N2CC3(NC(=O)Cc4ccon4)CCC2C3)=O)C1=O N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC(C2CC2)(CNC(C2CCCOC2)=O)C1 O=C(NNS(=O)(=O)C1CCCC1F)c1nc(C2CCC2)n(-c2ccc(F)cc2)n1 C1(NC(C(C)(F)F)=O)CN(C(C2CCCC(F)(F)CC2)=O)CC2CCCC12 CN1CCN(CC(=O)NC2(C(=O)NOCCCN=[N+]=[N-])CCN(C)C2)CC1 C(=O)(CS(=O)C(F)(F)F)NC1CCC(NC(NOCCC)=O)C1 N1(C(C2CCCCN2C(c2ccc(Cl)cc2)=O)=O)CC23CCC2(COC3)C1 CC1(CS(C)(=O)=O)CN(C(=O)C=CCC2CCCC2)C1 n1(CC(=O)N(C(C)CNC(C2CCCN(C)C2)=O)C)nc(C2CC2)n(C)c1=O c1(C(=O)NCCC2N(C(CCSCC)=O)CCOC2)sc([N+](=O)[O-])cc1Cl C(N=c1cc(NC(=O)NCC23CCCC2C3)nc(SC)[nH]1)c1cccc(CC)c1 C(=O)(C1=NOC(C)C1)NCCC(CNC(C1CCCN1N=O)=O)OC CC1(C)CCC=C1C(=O)N1CC2CC(C1)C2NC(=O)CCS(C)(=O)=O N1(C(CC2(C)CC2)=O)CCCC1Cn1cc(C2CC(F)(F)C2)nn1 CCC(CC(=O)N(CC(C)(C)CO)C1CC1)NC(c1ncccc1N)=O Cc1cncc(C(=O)N(C(C)CCNC(C2CC2c2cccnc2)=O)C)c1Cl N1(C(C)=O)CCCC1C(=O)NCCOCCNC(C1CC=CCO1)=O C(CCN=C(NCc1ccco1)NCC1(C#N)CC1)OC(C)=O.C(C)(C)(C)O C1(NC(CCc2cnc(C)o2)=O)CC12CCC(NC(C1(C)CCCOC1)=O)CC2 CS(=O)C1(CCNC(=O)N2c3ccc(s3)C2C2CC2)CC1.C(C)(C)(C)OC(=O)NC C(=O)(C(C#N)C(C)(C)C)N1CC(CC(=O)N(CC(C)(C)O)C2CC2)OCC1 Cc1ccc(C(=O)NCC2(C)CCN(C(=O)C3=CCCC3)CC2)c2c1CCC2 c1(C)cc(Cl)c(F)cc1F.CC1(C)CN(CCC(N2CCC(N)CC2)=O)CCS1 CC1CN(C(c2cc(C(F)F)on2)=O)CCCN1C(c1ccc(C(N)=O)s1)=O CN(C)S(=O)(=O)N(C)CC(N1CC2(CCC2NC(=O)CN2CCCS2(=O)=O)C1)=O C#CCC(C)(C)C(c1nnnn1CC1CC1)NCC(c1ccc(F)cc1F)CO CC1C(NC(c2cc(C3CC3)no2)=O)CCN1C(=O)C(c1ccccc1)=O N1(C(C(=O)N(CC(=O)OC)C(C)C)=O)CCC(C(=O)OC(C)(C)C)C(O)C1 c1(OC)nc(C)cc(C)c1CNc1ccc(C)c(SC(C)C)c1 C=CCC1CNC1=O.C1(O)(CC(=O)NC2CC(OCC)C2)CSC1 c1(C(N2CC3CCN(C(CC(=C)C)=O)CC32)=O)cc2c(SC)cccc2[nH]1 N1(C(C2(CNC(=O)NC)CC2)=O)CCOc2cc(Cl)ccc2C1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(c2ccc(C#N)cc2)=O)C(C)C1C Cc1cc(CNC(C2(CNC(=O)CN(C)C(C)C)CC(C)(C)C2)=O)cnc1C c1(NC2CC(CNC(CN3C(=O)CN(C)C3=O)=O)C2)nc(Cl)nc2c1ncn2C CC1(NC(c2csc(CNC(C3CC(=O)C3)=O)c2)=O)CC(F)C1 N1(C(C2CCN(C(C3(OCC)CCOC3)=O)C2)=O)CCCC2(CCC2)C1 C(CC(O)C(=O)NCC(O)CN(C(=O)C(C)(C)C1CCOCC1)C)SC CC(C#N)N(C)C(=O)NC(C)C1CC1 C(CCC(C)CC(=O)N1CC2CN(c3ncc(C)c(C(C)C)n3)CC2C1)=C(C)C C1(NC(c2ccc(C)cc2)=O)CN(C(c2nc(O)sc2C)=O)CC2(CC2)C1 C12(C(N(C3CCN(C(c4ccsn4)=O)C3)CCO)=O)CCC(F)(CC1)C2 CC1=C(C(=O)NC2CC3(C2)CC(C(=O)NC2CCSC2)C3)COCC1 C(=O)(C(C(C)NC(c1csc(Cl)c1)=O)C(C)C)NCc1ncc(CC)o1 C(CC(=O)NC1CN(C(=O)CCOc2ccccc2)CC12CC2)(C(F)(F)F)OC N1(C(c2c(CCC)n[nH]c2)=O)CCC(OCCCNC(c2coc(O)c2)=O)CC1 C(=O)(C1=CC2(CCOC2)C1)N1C(C(=O)NCC(C)C2CCC2)(C(C)C)CCC1 N1(C(=O)C=CC(F)(F)F)CC2(C(=O)NC3CC(CO)C34CCC4)CC1CO2 c1(C(=O)NC2CCC(NCc3cc(Br)ccc3O)C2)cccc2cc(Br)ccc12 C(=O)(N=c1nnn(C)[nH]1)N(CC(C)C(=O)Nc1cccc(Cl)c1)CCO c1(CNC(c2cccnc2)=O)nocc1C(=O)NCc1cccs1 Cc1ncsc1C=CC(=O)NC1CC2C(NC(=O)COc3ccon3)C2C1 C1(C(=O)NCCCC(C)NC(c2nc(CCCC)sc2)=O)SC2C=CC1CC2 Cc1[nH]cc(C(=O)NC23CCCC2N(C(=O)C=C2CCC2)CC3)c(=O)c1Cl C(=O)(CC(CC)C(C)(C)C)NC(CCCNC(C1CC(O)(CC#C)C1)=O)CCC C1(C(=O)NC(CC)(CC)CCNC(=O)CN(C)CCO)CCn2ncnc2C1 CC(C)(C)CCCCNC(C1CN(C(=O)CC2CCCNC2=O)CCO1)=O N1(C(C2NC(=O)OCC2)=O)CC2CC1CN(C(=O)Cn1cc(Cl)cn1)C2 c1(OC)ccc(C(=O)NCC2CC2CNC(C2CCC(C)O2)=O)c(C(F)F)c1 c1(NC2CCCC(NC(C(CO)NC(N)=O)=O)C2)nc2cc(Br)cnc2s1 C1(NC(C(C)OC(C)C)=O)CCN(C(=O)COc2cccnc2)CC1(F)F c1(OCC#C)ccc(C(=O)NCC(C2CCCC2)NC(C2COC(C)C2)=O)cc1 c1(NC(c2ccco2)COC)ccc(S(=O)(=O)NC2CS(=O)(=O)C2)cc1C#N c1(OCC(N2CC(C)(CNC(=O)CNC(=O)C3CC3)C2)=O)c(F)cccc1F Cc1cc(-c2ccc(N3CCN(C(=O)C(C)C4CC4)CC3)cn2)cnc1O.C(C)(C)O c1(CC(CC)C)nc(-c2cc(-c3ccccc3)cnc2)n(-c2nc(Br)nn2C)n1 N1(C(C2C(CC)C2)=O)CCC(O)(CN(C)C(c2ccn(CCF)n2)=O)C1 C(=O)(CCCCC(F)(F)F)N1C(CNC(=O)C=Cc2ccccn2)CC1 C(=O)(CC(C)CC(C)(C)C)NCC1OCCN(C(C(c2ccc(CC)s2)=O)=O)C1 c1(C(=O)NC(CNC(c2c(C)cccn2)=O)C)nc2ccccn2n1 CCCC(C(=O)NCCNC(C12CCC(CC1)C2)=O)C(C)C.c1ccnc(C)c1O Cc1cc(C(=O)N(CC(=O)NC(C)C(C)(C)O)C)ncn1 C(C(C)(C)C(=O)NC1CC1CNC(C1(C(F)F)CCCC1)=O)N(C)C c1(C(=O)NCCN(C(=O)CCC(F)(F)F)CC)cc2n(c1)CCOC2 N1(C(C(CCC)NC(C)=O)=O)CCC(NC(c2cn(C(C)(C)C)nn2)=O)C(C)C1 S(=O)(=O)(c1cccnc1NCCc1nccnc1C)NCC(C(F)(F)F)OC c1(C(=O)NC2CCN(C(C(CC)C(C)C)=O)C2C)ccc(OC)c([N+](=O)[O-])c1 C1(CNC(N2C(C(=O)OC)CC2)=O)(CN2CCCC2)CC(F)(F)C1 C1(OC)CN(C(c2cnccc2Cl)=O)CC1NC(=O)CCSc1nccn1C Cc1ccc2c(c1)CCN2C(C1CC(C)N1C(=O)CC1CCC(=O)N1)=O c1(-c2cccc(OC)c2Cl)cnc2ccc(C(N3CCNC(=O)CC3)=O)cn12 C1(C)(CNC(C2(C(=O)OC)C(=C)CC2)=O)CCN(C(c2ccno2)=O)CC1 CCC(CC)C(=O)NCC1(C2CC(NC(c3cc(-c4ccco4)c[nH]3)=O)C2)CC1 CN1CC2(CC2)CC1C(=O)NC(C(=O)NCC1(CC2CCC2)CC1)C1CCCO1 N1(C(CSc2c(OC)cccc2)=O)CCC(C2CC2)C1CNC(=O)CC(C)C C(CCC)(C(=O)NC1CCCC1CC(=O)N(C1CCNC1=O)C)=CCC CN1C(=O)CN(CC(=O)NCC2CCN(C(=O)CO)CC2)C1=O.C(C(F)(F)F)CO S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NC1C=CC(C(=O)Nc2ccc(C#N)nc2)C1 CC1CC(NC(=O)CSc2ccccc2Cl)CN1C(c1ccncc1Cl)=O N1(C(c2nc(C)[nH]n2)=O)CCCC(C2CC2NC(C2(C(F)F)CC2)=O)C1 CCCC(CC)CCC(=O)N1CCC(NC(C2(c3ccnc(Cl)c3)CC2)=O)C1C Cc1nn2ncc(C(=O)NCCCC3CCCCN3C(=O)C(C)SC(C)C)c2s1 c1(C(N(C(C)CNC(C23CCC2C3)=O)C)=O)cccc(C(N)=O)c1 Cc1cccc(C(=O)NN2CC3CCC3C2)c1.c12cc(n(C)n1)C(=O)NC2 c1(NC2CC3(C(F)C3)C2)nc2c(c(=NC3COc4ccccc4C3)[nH]1)CCCCCC2 c1(NC(C(C)NC(CN(CCC)C(C2(CO)CCC2)=O)=O)=O)cccn1C N1(C(C(COC)C)=O)CC(O)CC1C(=O)NC(C(C)C)C1CCC1 N1(C(COCC)=O)CC23CCCC2(C1)CN(C(c1n[nH]c(C)n1)=O)C3.C(=O)OCC c1(CCC)n[nH]c(=NCCCNC(c2ccc(OC(F)F)cn2)=O)s1 c1(C(c2nnnn2CCCC)NCC2(CCC=C)CC2)ccc(NC)c(OC)c1 N1(C(C2(C#N)CC(C)C2)=O)CCC(C(F)(F)F)C(NC(c2ccncc2)=O)C1 C1(C(N2CCC(C)C(O)C2)=O)(OC)CCN(C(=O)CSc2noc(C)n2)CC1 N1(C(c2cn(CCC)nn2)=O)CC2C(C(=O)NOCCOC)C2C1 c1(C(=O)NCC2C(NC(c3c(C)nc(O)cc3)=O)CC2)ncnc2c1CCC2 C1(C(=O)NCC2CC(NC(c3c(C(C)C)ocn3)=O)C2)CC2CCC1C2 N1(C(c2c(OCCC)cccc2)=O)CC2CCC1C1CN(C(C3CC3C)=O)CC21 CC(CC(F)F)C(=O)NCC1CCCN1C(=O)CSC1CCCCO1 N1(C(C(C)O)=O)CC2(CCC(NC(c3cc(Cl)cc(Cl)c3O)=O)CC2)C1 c1(CC)cccc(C(=O)NC2CN(C(=O)C(C3CCOCC3)F)CC2F)c1C CCC(C#N)C(=O)N1CCC(C(=O)NCc2nc(C)c(C)[nH]2)(CO)C1 c1(CC(N2CCC(C(CC)C)C2)=O)c(C)nc2ncnn2c1C.C1(=O)CN1CC c1(NCC(C)(C2CC2)NC(c2cnc(SC)nc2O)=O)nc(CO)nc(C)c1Br c1(Nc2cc(NCC(CCSC)OC)ncn2)ccc2nnc(C)n2c1 C1(CC)CN(C(=O)COC2CC2)CCC1NC(c1ccncn1)=O N1(C(C=COCC)=O)CCN(C(=O)C(Cc2ccccc2)NC(C)=O)C(CC)C1 C1(N2CCC(NC(c3cn(C)nn3)=O)C2)CCN(c2cccc(F)c2)C1=O C1(C(=O)OC)CCC2(CCN(Cc3ccc(C#N)c(N)c3)C2)C1 Cc1nccn1CC(N1CCCC1C(C)NC(C1(C(N)=O)CC1)=O)=O Cc1ccc(F)cc1C(=O)NC(C1CN(C(c2cc3sccc3[nH]2)=O)C1)C C(CCC(O)C(=O)N1CCN(C(C)=O)CC1C)NC(COCCOC)=O C1(C)(CNC(CCCOCC)=O)COCCN(C(C2CCS(=O)(=O)C2)=O)C1 C1(NC(CC2ON=C(C)C2)=O)CC2CC(C1)CN(C(=O)C1CCc3snnc31)C2 Cc1cccc([N+](=O)[O-])c1C(=O)NC1CC1CNC(=O)C=C1CCCC1 C1(NC(CC(C)C2CC2)=O)CC2CN(C(C3CCCCC3(C)C)=O)CC2C1 c1(C(N2CC(O)(CCNC(C(C)SCC)=O)C2)=O)ccc2c(O)nnc(O)c2c1 c1(C(N(C2CCCC2)CCNC(c2c(C)cc(C)o2)=O)=O)ccc2sncc2c1 Cc1c(Br)ccc(F)c1C(=O)NC1CC1CNC(c1cccc(C(N)=O)c1)=O CCCC(C)(O)C(=O)N1CCOC(C(=O)N(c2ccc(OCC)cc2)C)C1 CCC(CC)(C(=O)N1CC2CC1C2CNC(C1(C)CCCS1)=O)c1ccccc1 C1(CSCC)CCOC(=CC(=O)N(CCOCCCNC(C=CCC)=O)C)C1 N1(C(COC(C)=O)=O)CCC(NC(C2CC2c2ccccc2)=O)C1 c1(C(=O)NCc2cn(Cc3c(C(N)=O)cco3)nn2)cc2cccnc2[nH]1 CCCCC(O)CC(=O)N1CCCOC(CNC(c2cc(OC)nc(Cl)c2)=O)C1 N1(C(C(C)(C)NC(=O)OC)=O)CCCN(C(c2ccc(=O)n(C)n2)=O)CCC1 c1(C(=O)NC(CCCNC(C2(CC)CCCC2)=O)(C)C)c(Cl)sc(C)c1C N1(C(c2c(C)coc2)=O)C2CCC1C(C)C(NC(c1nc(C3CC3)cs1)=O)C2 C1(S(C)(=O)=O)(C(N2CCC(NC(C3(C)COCCO3)=O)C2)=O)CCOCC1 c1(CNC(CCC#C)=O)cc(C(=O)N(C2CC2(F)F)C2CC2)n(C)n1 C1(CC(=O)NCC2C(NC(CCN(C)CC)=O)C2)CSc2ccccc2O1 c1(CCN(c2snc(C)n2)C)ccc(Cl)cc1Cl C(=O)(CC(CC)CC(C)C)N(C(C(N1C(C(CC)O)CCC1)=O)C)C O=C(C1=CNC2=NCCCC2=C1)NCC1(F)CC(CNC(c2ccon2)=O)C1 C1(Cc2cn(C)nc2)CCCN(C(C(=O)Nc2ccc(F)cc2)c2cccs2)C1 C1(OCC)CC2(C1)CC2C(=O)NCC1(O)CCN(C(c2csc(Cl)c2)=O)C1 C(=O)(CC(C=C)CCC)NC(C(=O)NC(C#C)C(C)C)(C)CO C1(C(=O)NC(CO)CCO)(CNC(c2cc[nH]n2)=O)CC12CCC2 S(=O)(=O)(c1cccc(Br)n1)Nc1cncc(NC(=O)Nc2c(C)ncnc2C)c1 c1(C(N(C(C(N2CC(C=C)C2)=O)CC)C2CC2)=O)ccc(COC)cc1 N1(C(CCCN(C)C)=O)CCC(NC(C2CCC2)=O)C(CO)C1 c1(C(N2CCC(NC(=O)NCCC(=O)OC)C(F)C2)=O)c(C)cc(O)cc1C N1(C(C(CCCC)F)=O)CC2(CCC2)CC1C(=O)N(C)CCN(C)C1CC1 C12(CC(N3C(c4ccc(OC)nc4)CCC3)=O)COC(C)(C1)C2 CC1CN(C(c2ccoc2)=O)CC(C)N(C(C2CCN(S(=O)(=O)C(F)(F)F)C2)=O)C1 N1(C(C(C)=CC)=O)CCC2(CC1)CN(C(=O)Cn1nc(C)n(C)c1=O)C2C(C)C CC(=O)C(C)CC(C)C(=O)NC(CC1CC1)C(=O)NC1CC(CCC(N)=O)C1 C(=O)(C1CCCc2scnc21)NC1CN(C(C2C(C)=C2)=O)CC2(C1)CCC2 Cc1ccc2c(c1)C(CC(=O)NC1CN(C(=O)C(Cl)=CCl)CCC1(C)C)C(=O)N2 c1(C(=O)NCCCN(C(c2ccc(O)nc2Cl)=O)CC)cnc2ccnn2c1N N1(C(C(CC)C)=O)CCCC2(NC(=O)C=Cc3ncc(C)[nH]3)CC2C1 c1(C(=O)NC)cc(C)ccc1N(C)C(=O)NCCCNC(=O)COCCF N1(CC(C2CCOCC2)OC)CCC(=O)N(Cc2cc(OC)ns2)C1=O c1(C(=O)NC2(C)CCN(C(c3c(C)c[nH]n3)=O)C2)cnc(OC(C)C)c(Cl)c1 CCCC(C(=O)N1CCC2CC12C(=O)NC1(C)CC(N(C)C)C1)NC(N)=O N1(C(CSCCC)=O)CCC2(CC1)CCN(C(=O)CCF)CC2 Cc1cccc(CCC(=O)NC2CC(O)(CNC(C3(Br)CC3)=O)C2)c1 Cc1cc(C(=O)NC23COC(CNC(C45CCCCC4C5)=O)(C2)C3)c(C)cn1 CC(CC(=O)NC1(CCNC(C2CC23CC3)=O)CCC1)CC(C)(C)C c1(C(N2CCC(C(C)NC(c3cc(C)nc(O)c3)=O)C2)=O)cnn2ccn(C)c12 C(CS(=O)(=O)Cc1ccc(C)cc1)N(C(C1(COC)CCC1)=O)C Cc1cc(C)c(C=CC(=O)NC23CC(CNC(=O)CNC=O)(C2)OC3C)cc1C C=CC(C)(O)CC(=O)N1CCCC(C(=O)NC(CC)C(C)CN(C)C)C1 C(c1cccnc1)=CCNC(C(C)N(C(C(C1CC1)OC)=O)C)=O C1(C(=O)NCCCCCCNC(c2cc(C3CC3)no2)=O)Cc2nncn2C1 c1(SC)cccc(C(=O)N(CCCNC(C2CCOCC2(C)C)=O)C)c1[N+](=O)[O-] C1(C(=O)NC(CC#C)(C)C(=O)N(CC(F)F)CC)CC(=O)CC12CCC2 c1(C(=O)NC(CNC(CCc2cnc(C)s2)=O)(C)C(C)C)cc(Cl)cnc1O CC1(CNC(=O)CO)CN(C(C2CC(=O)C23CCC3)=O)CCO1 C(CC(=O)NCC12CC(CCO1)C2)(C(F)F)NC(c1c(C(C)C)occ1)=O C1(CNC(N(CCCCCC)C2CCCSC2)=O)CC2(C1)OCCO2 C1(C)(C(=O)NC(C)CN(C)C(c2c[nH]nc2-c2ccco2)=O)COC(C)(C)OC1 CC1CC(CC(=O)NC(CNC(C2(O)CCCC(C)(C)C2)=O)C2CC2)CC(C)(C)C1 C1(F)(C(=O)NC2CC(C)(CNC(c3ncc(OC)cn3)=O)C2)CCS(=O)(=O)C1 c1(C)cn(CCC(=O)CC(C)N(C)C)nn1.c1(C(NC)C)cnn[nH]1 C1(CC2CCN(CC(=O)N(C(C)(C)C)CCO)C3(C2)CC3)CC[Si]2(CCCC2)CC1 CCCCC(CNC(=O)C(C)OC)NC(c1csc(C(F)(F)C(F)(F)F)c1)=O C1(c2n(C(C3CCC3)NCCc3ccccc3F)nnn2)(SC)CCSC1C CCCCS(=O)(=O)CC(=O)NC1CC(CNC(=O)COC(C)(C)C(F)(F)F)C1 C12(C(=O)NCCC=C=C)CCN(C(=O)CCC3CC3C)CCC1C2 Cc1nc(CCC(=O)NC2CC(CNC(c3nnn(C)c3C(F)F)=O)C2)oc1C N1(C(c2c(OC(F)F)scc2)=O)CC2CC2C1.C(=O)(CC(C)c1ccncc1)OC Cc1nc(C)c(C(=O)NC2CC(N(C)C(C3CC3CF)=O)C2)s1 Cn1cc(C(=O)NCCN2CCN(C(C3(C#N)CCC3)=O)CC2)c(Cl)n1 Cc1nn(C)c(O)c1N(CC(N)=O)CC(N1CCOCC1)=O CCCC(CCO)NC(=O)C(C1CCN(C(c2ccnn2CCC)=O)CC1)C C(C1CCOC1)=CC(=O)NCCC1CCCN1C(=O)C=C1CCOCC1 c1(C(=O)NC2C(OC)CN(C(c3cc(C)nn3C)=O)C2)cc([N+](=O)[O-])cn1C c1(NC2CC(CC(=O)NCc3ncsc3Br)C2)ncc2cc(Br)cnc2n1 C12(NC(CSS(C)(=O)=O)=O)CCC(CN(C(c3cccc4nc[nH]c34)=O)C1)C2 C(C(C(=O)NCC1COC(=O)N1)NC(=O)Cn1ccc(C)c1)OC c1(C(N2C(CNC(CC=C(C)C)=O)CCCCC2)=O)ccc2c(c1)CCCO2 c1(NC(C#CCNC(C2(C=C)CCCC2)=O)=O)ccc2nc[nH]c2c1 N1(C(C(C)NC(C)=O)=O)CC2CCCCC2(CN=c2nc(C(C)C)[nH]s2)C1 N1(c2c(F)cnc(C)n2)CCc2c(CNC(C3CCOC3(C)C)=O)cccc2C1 CC(=O)CCCC(=O)NCC1CC1CNC(=O)CCCc1nc(C2CC2)no1 N1(C(CC2CC(OC)C2(C)C)=O)CCC(Nc2ncnc(O)c2Br)C(C)C1 CCN=c1[nH]cc(C(N2CCC(CCNC(=O)CCOCC(C)C)C2)=O)s1 C(CCCCNC(=O)CC1CCC1(C)C)NC(CCN(CCC(C)(C)C)C)=O c1(CN(CC=C)C(=O)NC2CCN(c3ccncn3)CC2)ccc([N+](=O)[O-])cc1 C(=O)(C1CCCc2c[nH]nc21)N1C2CC(NC(C(CCCC)N(C)C)=O)(C2)C1 c1(C(=O)NC2CC(F)(CNC(c3n(CC)ccc3)=O)C2)ncc(Cl)cc1Cl C1(C(=O)NC2CCCC2NC(=O)C(=CC2CCCC2)C)(COC)CC=CC1 c1(C(=O)NC(C(C)NC(c2cc(C(N)=O)[nH]n2)=O)CO)cc(N)ccc1Cl c1(C(N2CCC(N(CC)CC)C2)C(=O)NC(C)C)ncc(C(C)(C)C)cn1 CC(C(=O)NCc1cc(C(=O)NCC2CC23CCOCC3)ccn1)S(C)(=O)=O C1(C)(CNC(C(C)NC(CC)=O)=O)CCCN1C(c1cc(OC)ccn1)=O N1(C(C(CC)C(C)C)=O)CC2CCOC2(CNC(=O)CCC(=O)N(C)C)C1 C1(C(N(CCNC(C(N2CCCCCC2)C)=O)C)=O)C(O)C(=O)N(C)C1C C1(C(C)NC(C=CC(C)C)=O)CN(C(c2ccnn2CCF)=O)CCO1 C1(C(=O)NC(c2ccncc2)C)CC1C1CN(C(=O)C(C)(C)C(C)O)C1 CCC(COC)(CC)C(=O)NCC1CN(C(C2COC(=O)N2C)=O)C1 C(=O)(CC(=O)NC(CNC(c1c[nH]nc1C(F)(F)F)=O)CO)N(C)C c1(OC)ccc(C(=O)NC2CC(Nc3ccn4ncc(I)c4n3)C2)cc1[N+](=O)[O-] C(C1=CCC2CC1C2(C)C)(c1nnnn1C1CCCCC1)SC.C1CN1CCI C1(C2CN(C(=O)CCc3cccc(O)n3)C2)(NC(Cc2c(C)n(C)nc2)=O)CC1 CC(C)C(C)(C)C(=O)N1CCC(NC(=O)CC2CC(=O)NC2=O)C(C(N)=O)C1 c1(CC)[nH]nc(Cl)c1C(N1CCC(CO)(NC(c2cc(C#N)c[nH]2)=O)C1)=O C(C)(C(=O)NCCN(C)CC)(C1CCC1)NC(C(C)O)=O.C#CCCC C1(C(N(CCC(C)NC(=O)CCCOc2ccccc2)C)=O)CCC(=O)N1 S(=O)(=O)(c1ccc(NCCS(C)(=O)=O)cc1Br)N(C(F)(F)C(F)(F)F)C n1(C(CN(C(CC(C)C)C(=O)NCC(C)C)C(N)=O)C)cnc2ccccc12 C1(N(C(Cc2cccc(OC)c2)=O)C)CCN(C(C2CC3CC3C2)=O)CC12CC2 C1(C2CC2)(CNC(C(c2cccc(C)c2)O)=O)CCN(C(=O)CC(C)N(C)C)C1 C1(C(=O)NCC2CCC(NC(=O)C(C3CCCCC3)O)C2)CCCCCC1 C(=O)(C1=CS(=O)(=O)CCC1)N1CC(C(C)NC(c2c(C)cno2)=O)C1 C(=O)(C(CCOC)NC(c1ccc(C#N)cn1)=O)OCCC c12c(cccc1C)S2.c1(OC)ccccc1CC12CC(C(=O)OC)(C1)C2 C(CC(C(=O)O)N(C(=O)Cn1cc(CNC(c2ccccc2N)=O)nn1)C)SC CC1=C(C(=O)N2CC(C3CN(C(c4cnc5sccn45)=O)C3)C2)CCCC1 c1(C(N2C(CNC(C3(OC)CS(=O)(=O)C3)=O)CCC2)=O)cccn2cnnc12 c1(-c2ccc(C(=O)Nc3nc4ccccc4[nH]3)nn2)cnc2[nH]cnc2c1 N1(C(C2N(CC(C)C)CCC2)=O)CCOC(C)(CNC(C2CC3CC3C2)=O)C1 CCCCCCC(=O)N1CC(F)CC1CNC(C1(C)CC2(CCC2)C1)=O c1(C(C(=O)NCCC2CC(NC(c3c(C)nns3)=O)C2)N(C)C)ccc(Cl)cc1 CCC(C)CCC(=O)NC1COCCN(C(=O)C(c2cccc(Cl)c2)(C)C)C1 Cc1nc(C2CC2)nc(O)c1C(N1CCOCC(NC(C2(C)CCCC2)=O)C1)=O c1(OCC(=O)NCCC2CCN(C(=O)C3=CCC3)C2)cccc(F)c1F C#CC1CN(C(=O)CC(C)NC(=O)C(C)CC(=O)OCC)CCN1C C1(C(=O)NCCCOCCCNC(c2sc(C)c(O)n2)=O)CCCCNC1=O C1(C(N2CC(F)(F)C2)=O)CC2CC2N1C(=O)C=CC1CCOC1 Cc1cc(N2CC(CNC(=O)CCc3cn[nH]c3)CC2C)ccc1[N+](=O)[O-] c1(OCC)ccc(C(=O)NC2CC(CCNC(=O)Cc3cc(C)no3)C2)cn1.C1CC1 N1(C(c2ccc(C(CC)C)cc2)=O)CCCC(C)C1CNC(C1(CSC)CC1)=O C1(NC(CCc2cn(C)nc2)=O)C(C(=O)O)(OCCN)CC1(F)F O=S(=O)(c1cnc(NCC2CCC(F)C2)c(Cl)c1)N1CCc2cccnc2C1 c1(C(N2CC3C(NC(c4cccc(C)n4)=O)C3C2)=O)c(C)cc(O)nc1C Cc1ccc(C(N2CCC(CCNC(c3cc(C4CCCC4)no3)=O)C2)=O)cc1 C1(CC)C(NC(c2ccco2)=O)CCN1C(=O)C(COC)OC C1(NC(C(C)N(C(=O)C(C)=C(C)C)CCC)=O)CCOC(C=O)C1.OC c1(OC)cc([N+](=O)[O-])c(C(N2CC(CN(S(=O)(=O)CCCCl)C)C2)=O)cc1O Cc1cccnc1CCC(=O)NC(CN(C(=O)Cc1cnnn1C)C)(CO)CO CCC(CCC(=O)NCC(N1CCCC1)C)NC(=O)Cc1ccccc1F C1(NC(CCCC(C)C)=O)CN(C(=O)C=Cc2cn(C)cn2)C2(CCCOC2)C1 c1(C(N2C(CNC(C(CCC)NC(C)=O)=O)CCC2)=O)c(OC)ccc(F)c1N C1(CNC(=O)Cc2ccc(O)cc2)Cc2ccccc2CN1C(c1ccc[nH]1)=O c1(NC(N(C(C)Cc2ccsc2)C)=O)cccc(-c2ccnn2C)c1 N1(C(C2(C(C)C)CCC2)=O)CC2(CCCN(C(C3CC(=O)N(C)C3)=O)C2)C1 n1(CC)nc(C)c(C(N2CCC(C)(NC(=O)CC3CC(SC)C3)C2)=O)c1Cl C1(NC(c2cnc(SC)s2)=O)CC2CC1N(C(c1ccc(F)cc1N)=O)C2 N1(C(C2N(C(CCC(=O)OC)=O)CC2)=O)CCC(CC2CCCC2)C(O)C1 N1(C(C(CCSC)NC=O)=O)CCCN(C(C2(CF)CCC2)=O)CC1C c1(C(=O)NCC2CCN(C(C3CC(F)C3)=O)CC2)cc2c(cc1[N+](=O)[O-])OCO2 c1(C(=O)NCC(CNC(c2ccc(Cn3cccn3)o2)=O)F)ccnnc1S CC1(NC(=O)CC2CCC(O)C2)CCN(C(c2n[nH]c(=N)s2)=O)CC1 C(C(CNC(=O)COCC1CCC1)C(F)(F)F)NC(c1cccc(C)c1)=O c1(CC)cccc(C(N2CC3C(NC(=O)C=Cc4nnc(CC)o4)C3C2)=O)c1O c1(OC)ccc(-c2ccc(C(N(C3CC(=O)NC3=O)C3CC3)=O)cc2)cn1 N1(C(=O)CC23CCC(CC2)C3)CCC2CN(C(c3cc(O)cs3)=O)CC2CC1 CCCC(C)CNC(=O)C(CNC(C1(C)CC=CC1)=O)OC C(=O)(C(CSC)NC(=O)CCc1nc[nH]n1)NC(CC)CSC C1(CNC(C2N(C)CC(O)C2)=O)CC2(CC(NC(=O)CC3CC4CC4C3)C2)C1 N1(C(C2N(C(C(C=C)OC)=O)C(C)C2)=O)CCC(OC)CC1 CCCCCC(C)CC(=O)N1CC(C2CC2)(C(N2CCOC(C)(C)C2)=O)C1 N1(C(CCc2ncc(C)[nH]2)=O)CCC2(CC1)CCN(C(C1COCCN1C)=O)C2 Cc1nncc(C(=O)NCC(C)(C)CC(=O)N(C2CCCC(C)(C)C2)C)c1C N1(C(C2CC23CCSCC3)=O)CCC2C(C1)CN2C(c1cnn[nH]1)=O C(c1ccc(Cl)s1)=CC(=O)NC(C1N(C(C=CC=CC)=O)CCC1)(C)C N1(C(C(C2CCOCC2)C)=O)CSCC1C(=O)NC1CCCC1c1nc(S)n[nH]1 C(=O)(C1=CCCCC1P(C)(C)=O)N1CC(C)CN(C(c2ccc[nH]2)=O)C(C)C1 C1(C(=O)NC2C(OC)C(O)C2)CN(C(C2CC(CC3CC3)C2)=O)C2(CCC2)C1 C=CC(CC)C(=O)N1CCOC(CC(=O)NC2CCNC2=O)C1 C(=O)(C1=C(Cl)CCOC1)N(C)CC1CN(C(=O)C(N)=O)CCO1 C(C)(C)(C(C)CC(=O)NCC1(CCO)CCC1)NC(CNC(=O)NC)=O C(=O)(C(CN=[N+]=[N-])NC(=O)C(O)C1CCCC1)N(C)Cc1nccn1C c1(CC(C)NC(=O)C(C)(F)F)cn(CCF)nn1 O=C1CN(C(=O)C(C2(O)CCCCC2)NC(C2CC23CC3)=O)CC(=O)N1 C(=O)(CCCN(C(=O)CNC(C1CC1C)=O)C)NCCOC(C)C N1(C(C(C)SC)=O)CC2CC(NC(=O)C(C(C)C)C3CCC3)C2C1 C(=O)(CC(C)(C(F)(F)F)N(C)C)N1C(CNC(C(C)=CC2CC2)=O)CC(O)C1 CN1C(=O)CC(C(N2CC(F)(F)CC2CN)=O)C1c1cnn(C)c1 c1(OC)ccc2[nH]c(C(N3CC(CNC(=O)C(C)CN(C)C)C(C)C3)=O)cc2n1 C(=O)(C(C1CCCO1)N(C)C(=O)C1CC1)NCCN(CCC)CC CC1(C)COCCC1CC(=O)NCC1CCN1C(=O)C(c1ccc(Cl)cc1)CO CC#CCC(C(=O)NCc1n[nH]cc1CC)NC(c1cc(OC)no1)=O Cc1cc(=NC2CC3CCC2N(C(=O)C(F)NCC)C3)c(F)c[nH]1.OC(F)(F)F c1(C(=O)NCCC(CNC(C(CCC)N(C)C)=O)O)c(O)cc(Cl)cc1F C1(C2(O)CCC2)(C(=O)NC2CC(CNC(C=C(C)C(C)(C)C)=O)C2(C)C)CC1 c1(C2C(NC(CCN(C(C3(O)CCC3)=O)CC)=O)C2)ccccn1 c1(C(C(=O)NCC2OCC(CNC(Cc3c(C)non3)=O)C2)=O)ccc(O)cc1 n1(CCCC)nnc(C(=O)NC2CCN(C(c3cnc(S)n3C)=O)C2)c1C N1(C(C23CC(NC(CC4C(C)CCCO4)=O)(C2)C3)=O)CCC2CCCC2C1 C1(CCOC)(NC(C2CC=CCC2)=O)CCN(C(c2cncs2)=O)C1 N1(C(c2c(CC)noc2)=O)CCC(CCNC(=O)C(C)OCC2CCCO2)CC1 C1(O)(C(C)NC(=O)CCc2cccnc2)CCN(C(=O)C(F)(F)C(F)F)CC1 N1(C(Cc2ccc(F)cc2F)=O)CCC(C2CN(C(c3c(C)ccs3)=O)C2)C1 c1(NC)cncc(C(N2CCC(NC(c3ccoc3Br)=O)C2C(C)(C)C)=O)c1 CCC(C)C(=O)NCCC(Cc1ccccc1)NC(c1sccc1C)=O c1(-n2ccc(C)n2)ccccc1C(C1CC1)NC(=O)NCCN1CCOC(C)C1 c1(C(=O)NCC(CNC(c2ccc(C(C)=O)nn2)=O)(C)C)cc(Cl)cc(C)c1C c1(NC(=O)COc2ccccc2OC(F)F)nccc(N2CCCCC2)n1 CC#CCCCCNC(=O)C(CC=CC)NC(=O)Cc1cc(C)[nH]n1 Cc1nc(S)sc1CC(N1CC(NC(C2(O)CCCCC2)=O)C(C)C1)=O c1(C(=O)NCCCC(F)F)ccc2c(c1)CCOC2 C(CCCC(=O)N1CCC1(C)CC(=O)NC(c1ncccc1F)C)OCC C(=O)(C(CC(C)C)OC)N1CCC(CC=C)(NC(c2oc(C)cc2C)=O)C1 c1(CC)ccc(C)c(C(N2CCN(C(C34CC3CCC4(F)F)=O)CC2)=O)c1 CCC1=C(C(=O)N2CC(NC(c3cncnc3C)=O)C3(CCC3)C2)CCCO1 C1(C(=O)NC(CC#C)C(=O)NCCNC(=O)C2CC2)CC2C(C1)C2(F)F c1(NCC(=O)NC2(CNC(C3C(C)C3)=O)CCOC2)cncc(C(F)(F)F)c1 C1(N(c2c(C)coc2)C(=O)C(C)C)CC2CCC1CN2C(=O)CC(=O)N(C)C n1(CCC)cc(Cl)c(C(=O)NC2(CO)CN(Cc3ccc(Cl)cc3)C2)n1 c1(CCC)ccc(N)c(C(=O)NCC2CC(C)(C)CN2C(C2CCOC2)=O)c1 Cc1nn(C)c(C)c1C(N1CCN(C(C2(C)CC3(CC3)C2)=O)CC1)=O C1(C(N2CCC(NC(Cc3ncc(C)[nH]3)=O)CC2C)=O)CCc2cnc(C)n2C1 C(C(=O)N(CC(=O)NCC(C)C)CC(C)C)(C1CCOC1)NC(C)=O c1(C(C(=O)NC(CC)C)N(C2CCN(C)C2)C)ccc(OC)c(C)c1C Cc1ccc(-c2cn(C(C)C(=O)NC(CO)CC(C)(C)C)nn2)cc1C#N c1(OC)ccc(-c2cnc(NC(c3n[nH]cc3[N+](=O)[O-])=O)c(C)c2)c2cn[nH]c12 N1(C(C(C)c2cncs2)=O)CC(O)CC1(C)C(=O)N(C)CCC1CC1 N1(C(c2ccncc2)=O)CCCC(S(=O)(=O)N2CCc3sccc3C2)C1 C1(NC(CSCC)=O)CN(C(=O)CCCOC(C)=O)CC2(CC2)C1 C1(C(N(C)CC2CN(C(c3ccns3)=O)CCO2)=O)CCCC2CCCN12 N1(C(c2c(OC)cccc2C)=O)CCC(C)N(C(=O)CSc2n[nH]c(O)n2)CC1 c1(C(N2CCC(NC(c3c(Br)ccc(C#N)c3)=O)C2)=O)cc2c(cc1Br)OCO2 N1(C(=O)COC2CCCC2(F)F)CCCC2(C1)CN(C(C1CCOC1)=O)CCO2 c1(C(N2CCN(CCCNC(=O)C(F)(F)C3CC3)CC2)=O)csc2nnsc12 C1(NC(c2scc(C)c2)=O)CCN(C(=O)CCCCCNC(N)=O)CC1C C1CCC(C2(Nc3ccc4sncc4c3)CCNCC2)CC1 Cc1nc(-c2ncc[nH]2)sc1C(=O)N(C1CCCN(C(=O)CS(N)(=O)=O)C1)C N1(C(=O)OC(C)(C)C)CCn2c(Br)cnc2C1.c1(C(C(=O)N)NC)cccnc1 c1(C(CNC(C2(C3CCCCO3)CC2)=O)NC(=O)C=CC2CC2)ccc(F)cc1 C(C1(O)CCCc2ccccc21)NC1CC2(C(OC)(OC)CC2)C1 C1(O)(CNC(C2(C)C(CC)CCC2)=O)CCN(C(=O)CNC(=O)C(F)(F)F)CC1 C1(OC)(CNC(=O)CCF)CCN(C(=O)CC2CCCCN2c2ccncc2)C1 C1(c2cccc(OCC(F)(F)F)c2)(NCc2ncc(C)s2)CCOCC1 C1(NC(c2n[nH]c3c2COC3)=O)COCCN(C(c2ccnc(O)c2F)=O)C1 N1(C(=O)Nc2cccc(CSCC)c2)CC2CCCC2(CO)C1 Cc1ncc(C(=O)N(C2CCCN(C(=O)C(O)C3CC3)C2)CC2CC2)c(C)n1 CCCC(C(=O)NC1(C)CCN(C(=O)C(CO)c2ccccc2)C1)N(C)C Cc1ccc(F)c(CC(=O)NC2(C)CCN(C(c3cc(N)c(Cl)cn3)=O)C2)c1 c1(CC)cc(N)c(C(=O)N(CC(O)CNC(=O)COC(F)(F)F)C)cc1F c1(OC(c2ccccc2)C)ccc(NC(=O)CCc2cnc(Br)s2)c(I)c1 c1(C(=O)NCC2C=CC(NC(C3(CCCC)CC3)=O)C2)nc2nc(C)ccn2n1 C1(CN(C(C(=O)N(C(COC)C)C)=O)C)COCC1OC C1(NC(CCCc2nc(C)sc2)=O)CC(CO)N(C(C2COC(=O)C2)=O)C1 c1(NC(c2c[nH]ccc2=O)C)ccc(S(=O)(=O)N2CCCCC2C#N)cc1Br C#CC(CNC(=O)C=C1CC1CNC(=O)CC=CC=C)CC1CC1 C1(NC(C(CCC)(C)C)=O)CN(C(=O)C(F)n2cccn2)CC2(CCOCC2)C1 C(CC(C)(C)CNC(=O)C(C)(C)CC)NC(C(CC)N1CCCC1=O)=O C1(C(=O)NCC(CN(C(c2c(OC)n[nH]c2)=O)C)O)C2CC(=O)CC12 C1(NC2=NOCCN2C2CC(C)OCC2)CCOc2ccccc2C1 Cc1c[nH]cc1C(=O)N(CCC(C)NC(c1cnn(CC2CCC2)c1)=O)C C(=O)(N=c1cc[nH]c(C)c1C1CC1)c1c(C)nn(-c2ccc(S(C)(=O)=O)cc2)c1 N1(C(CCOC(C)=O)=O)CCC2(CC2C(=O)NC2CCCN(O)C2=O)C1 c1(Cn2c(C(CCC3COC(=O)C3)NCc3ccoc3)nnn2)ccccc1 Cc1nc2ncccn2c1C(N1CCSCC1C(N1CCCC(C#N)C1)=O)=O C(CCSC)(C(=O)N(C)CCN(C)C)NC(C(CC)SC)=O.C(C)(=O)N c1(CCN(C2CC23CCNCC3)C(CC=CCC)=O)c[nH]c2ncc(C)cc12 N1(C(C2C(CC)CCC2)=O)CC(C(=O)NCCCC(F)(F)F)CC12CCC2 Cc1n[nH]c(C)c1C(C)NC(C1CCCN(Cc2cncc(C3CC3)c2)C1)=O C(=O)(CCCN=c1nccc[nH]1)N1CC(SC)C(NC(C2CN(C)C2)=O)C1 CN1CCN(CC(=O)NC2CC(F)CN(C(c3ccc(C)n3C)=O)C2)CC1=O C1(OC)(OC)CC(C(=O)N(C)CCOCCN(C(=O)C(C)(C)c2ccno2)C)C1 c1(NC2(c3n(CCCOC)nnn3)CSC2)ccc(OCC(F)F)cc1 N1(C(C(C2CCCO2)NC(c2scc(C)c2)=O)=O)CC2(CCC2)CC1C c1(CO)ncc(C(c2cccc(C(=O)NC3CCCCC3C(=O)O)c2)=O)cc1Cl C1(CNC(C(CCOC)C)=O)CC2(CC2)CN1C(=O)Cc1occc1C c1(NCCC(=O)N(CCC)Cc2ccccc2)c(F)cc([N+](=O)[O-])cc1F CN1CCN(C(C2CN(C3COC3)C2)=O)C(C(N2CCC23CCCC3)=O)C1 C1(C(=O)NC(c2nnc(C)o2)C)CCC(NC(=O)C(C)C2CCCC2)CC1 N1(C(=O)CC2(CO)CCCC2)CC2CC1CC2CNC(c1cc(C2CC2)no1)=O N1(C(c2c(C)c(Br)ccc2F)=O)CCC2(CC1)CC2(C)C(N1CC2CC2(C)C1)=O c1(N2CCCC3(NC(c4cnc(C)o4)=O)C(C2)C3)nccc(C)c1[N+](=O)[O-] N1(C(C(C(CC)O)C)=O)CCC2(CCN(C(c3ccc(C)n(C)c3=O)=O)C2)C1 c1(C(N2C3CC(NC(C4(C(C)C)CC4)=O)C2CC3)=O)ccc2c(c1)CCN2C C12(C(=O)NC3CC(CCNC(c4cc(C(C)C)on4)=O)C3)CCCCC1C2 N1(C(CCC2(C)CCC(=O)N2)=O)CC2CCC1C2C(=O)NC1(c2cccs2)CC1 C1(NC(COC(C)(C)C)=O)C=CC(CC(=O)Nc2csc(Cl)c2)C1 c1(SCC(=O)NCC(C)NC(c2csnn2)=O)ccccn1 C(CCCC(=O)N1CCC(N(C(=O)Cn2nccc2C)C)C1)NC(C)=O N1(C(C(C)=C(CC)C)=O)CC2C3CCC(C2C1)N(C(=O)CC1CC2CC2C1)C3 c1(C(C)(C)C)cccc(Br)c1Br.CC(CSC)NC C(C(=O)N1CC2CC1CN2C(=O)OC(C)(C)C)(C(C)C)c1cccc(C)c1 c1(NC(CN(C(=O)C(c2cc(Br)cs2)O)CC)=O)nc(CC2CC2)cs1 c1(C(=O)NCC(CC)N(C(=O)C(n2ccnc2C)C)C)cc(O)nc(O)n1 C=CC1OCCC1N=c1nc(N2CCN(C)C(C(F)(F)F)C2)c2c([nH]1)CCOC2 C(CC(O)C(=O)N1CC(NC(c2ccc(NCC(F)F)nc2)=O)C1)N(C)C C1(C(N2CCC(SC)C2)C(=O)NC)CCC(n2ccnn2)CC1 CC(=NO)C1CC(C(=O)NCC(C(C)C)NC(c2c(C)cccc2N)=O)C1(C)C CC1CN(C(c2cnoc2)=O)CCC1NC(=O)Cc1cc[nH]n1 c1(CNC(=O)NCc2ccc(N3CCCC3)nc2)cccc(-c2ccccc2)n1 n1(CCC(=O)NC2(CNC(C(CC)CC)=O)CCOC2)cnc2sccc2c1=O N1(C(C=C(C)c2cnn(C)c2)=O)C2CCC1CN(C(=O)CN1CCSCC1)C2 c1(NC(C2CCCC(CNC(C(C)=C(CC)C)=O)C2)=O)sc(C)c(C)c1C(N)=O Cc1cc(S(=O)(=O)NC2CCC2O)n(C)n1 N1(C(c2cc(C)c(C)s2)=O)CC2=C(C1)CN(C(=O)CC(C)(C)C)C2 c1(CCC(=O)NC(C2CC2n2cc(-c3nccs3)nn2)C)cc(F)ccc1F CC1(C)CCCN(C(C2CCCS2)=O)C1C(=O)NCc1cnn(C2CC2)c1 C1(C(N2C(CCNC(=O)CC=C(Cl)Cl)CSCC2)=O)CCc2nnc(O)n2C1 c1(CNC(c2c(C)ccs2)=O)cc(C(=O)NCC(=O)OC(C)C)ccn1 C1(C(F)F)(CNC(c2nnnn2Cc2ccco2)c2ncco2)CCCC1 N1(C(c2cncc(N(C)C)n2)=O)CCC(C2CC(NC(=O)CC(C)(C)C)C2)C1 C(=O)(CCCCCCCO)N1CC(C)C(CNc2ccncc2[N+](=O)[O-])CC1 c1(C(=O)NCCCC2(NC(C(c3n(C)ncc3)=O)=O)CC2)cncc2nc[nH]c12 S(=O)(=O)(c1ccc(Br)cn1)NCCc1nc(COCC)on1 C(=O)(C1=CCC1)N(C(C)CCNC(=O)C(C)SC(F)(F)F)C CN1CCn2nc(C(N3CC(C4CCN(C(=O)C5CC5)CC4)C3)=O)cc2S1(=O)=O c1(C(=O)NCC2CC2NC(c2ccsc2C2CC2)=O)cc2ccc(Cl)cc2[nH]1 CCC(O)C(C)C(=O)N1CCC(C(C)NC(C2CCN2CC)=O)CC1 c1(OC)ccncc1C(=O)N(C)CC1CN(C(=O)CC(C)(C)C2CC2)CCO1 C(CCCCC(=O)NCCC1(C)N=N1)NC(C1(CSC)CCC1)=O c1(C(=O)OCC2(C)COC2)cc(Cl)nn1-c1cccnc1 c1(CC)ccc(C(C)C(=O)NCC2CCC2NC(c2c[nH]nc2C(C)C)=O)cc1 C(=O)(CC(C)C(F)(F)C(F)(F)F)NCC(C)N(C(c1c(COC)nn(C)c1)=O)C N1(C(C(=O)NCc2c(OC)cccc2)c2ccns2)CCCC(C2CCCC2)C1 c1(C(=O)NC2C3CN(C(C=C)=O)CC32)ccc(S(=O)CC#N)cc1 Cn1nccc(-c2ccc(C3CC3(C)C)cc2)c1=O c1(OCC)c(C(=O)NCC2(OC)CCN(C(C3(C)CC3)=O)CC2)cccc1F c1(C(CC)C(=O)N(CC(C)NC(c2ccn(C(F)F)n2)=O)CC)ccc(Cl)cc1 CC1CN(C(=O)CC2CNC(=O)O2)CCC1CNC(C1CC2(CC2)C1)=O n1(CC)ccc(C(=O)NCC(C)CN(C(=O)CC2CC23CC3)C)cc1=O C1(OC)CC(CNC(=O)C(n2cc(C)cn2)C)N(C(c2cccc(O)n2)=O)C1 N1(C(c2cnc(OCC)c(Cl)c2)=O)C2CCC1C(F)C(NC(=O)C(F)C(C)C)C2 CCC(C)(C)C(=O)C(=O)N1CCC(NC(c2cc(F)ccc2NC)=O)C(F)C1 C1(NC(c2ccc(CC)s2)=O)CCCN(C(C2CCCN2CC(C)C)=O)C1 c1(C(C(=O)NCc2c(CC)c[nH]n2)(F)F)ccc([N+](=O)[O-])cc1Cl N1(C(C(CC)Cl)=O)CCC2C1CCN2C(c1n[nH]c(C)c1F)=O c1(C(N2CCC(C)(CCNC(C(C)OCCCC)=O)C2)=O)ccnc2c1CCC2 C(C)(N=c1[nH]c(=NCCOCC(=O)OCC)c2sccc2[nH]1)=CCCC c1(C(c2nn(C)cc2I)N(C)Cc2nnnn2C)ccc(Cl)cc1 N12CCOC(C1)SCC2=O.C1(CC(=O)N(CC)CC)CCN(C(C)=O)CC1 C1(N(C(c2cnn(C)c2)=O)CC)CCN(C(C2(C(N)=O)CCC2)=O)CC12CC2 CC1CC(NC(C2N(C(C3CCCC3)=O)CCCC2(C)C)=O)CC1(C)C N1(C(C(C)CF)=O)CC2CC(C1)CN(C(c1cc(-c3ccccc3F)no1)=O)C2 C1(C(N(CC)CC2CCCN2C(C2CS(=O)C2)=O)=O)CCOC(C)(C)C1 CC(C)CCC(O)C(=O)NCCC(C)NC(c1ccc(CNC(N)=O)cc1)=O N1(C(COCC=C)=O)CCC2CN(C(=O)Cc3ccc(C)c(F)c3F)CCC2C1 C=C1CC2(C1)CC(C(N1CCCN(C(=O)C(C)NC(=O)OC(C)(C)C)CC1)=O)C2 C1(C(N2CCC(CC#C)(C(=O)NCC3CCCC3(C)C)C2)=O)C2CC3C(C2=O)C13 Cc1cc(C(N2CCC(OCCNC(C34CCCC3C4(F)F)=O)C2)=O)nc(C)c1 c1(OC)c(CC(=O)NC2CCCC2NC(c2cn(C)nc2C)=O)cccc1C#N c1(C(=O)NCC(C)N(C)C(c2cn(C)nn2)=O)ccc(C(C)(F)F)cc1 C(c1ccc(-c2ccccc2)s1)=C1CN(C(=O)CC2CC(O)CN2)C1 N1(C(C2CN(C(=O)NC)C2)=O)C2CCC1CC(C(=O)NCC(c1cnc[nH]1)C)C2 c1(NC(C2N(Cc3cnc(N(C)C)c(Br)c3)CCC2)=O)ccc2c(c1)CCCC2 N1(C(C(COC)OC)=O)CCC(CNC(c2cnn(C(C)C)c2N)=O)C12CC2 CCC(CN(C)C)CC(=O)N1CCCCC1CSc1cn(CCCCCO)nn1 C1(CNC(C(COC)CC)=O)CCC2CN(C(=O)Cc3sccc3C)CC12 C1(O)(CCNC(C(C=CC)O)=O)CCN(C(C2(C(C)(C)O)CCC2)=O)C1 C1(CC)CCC(C(=O)NCc2ncc(CO)o2)O1.C1(C)C=CC(=O)N1 C1(=O)CCCN(C)C(=O)C(CCCC(C)OC)C(=O)NCCCN1CC C=C(CN(C(=O)CCCN(C(=O)C(C)CCCOC)C)C(C)C)c1ccccc1 CCCCC(C)(F)C(=O)NCC1(NC(c2n[nH]c(C)c2C)=O)CCOC1 C1(O)(CNC(C(=C)F)=O)CCN(C(c2ccc(C)cc2)=O)C1 c1(C(C2(C(=O)NCC3N(C(=O)CF)CCOC3)CC2)=O)cnc2scnc2c1 CN1C2CCC1(C(=O)NCC1CC(O)CN1C(=O)CCn1cncn1)CC2 Cc1ccc(CC(=O)NCC2CC2NC(=O)Cc2cccc(Cl)c2)cc1 N1(C(c2nc(C(=O)OCC)oc2)=O)CCN(C(C23CCC2C3)=O)CC(C)(F)C1 N1(C(c2ccc(C)nc2)=O)CCCC(O)(CNC(=O)CC2CNC(=O)O2)CC1 c1(C(C)=O)ncc(C(=O)NC(C)C(CO)NC(=O)C(CO)c2ccccc2)s1 N1(C(CC(C)Cc2cccc(F)c2)=O)CCOC2(C1)CN(C(C1CCO1)=O)C2 c1(NC(=O)NC(C(=O)OC)C2CCCO2)ccc(Br)c(Cl)c1F c1(C(N2C(C3CN(C(C4C(OC)C4)=O)C3)CCCC2)=O)cccc2c1OCC2 C1(C(=O)NCCC(COC)(C)C)CN(C(=O)Cc2csc(C)c2)CC12CCC2 c1(C(=O)NCC2C=CC(NC(C3CC34CC4)=O)C2)cc(F)cc2nccnc12 C1(C(=O)NC2(C)CCC(C)C2)CC2CCC1N2C(C1CC2(C1)CC(O)C2)=O c1(N2CCC(N(C)Cc3cccs3)C2)ccccc1F N1(C(C2(C)CCN(C)C2=O)=O)CC2CCN(C(=O)Cc3ccc(Br)cc3)CC12 c1(C(N(CCNC(=O)C(F)n2cccn2)CC)=O)ccc2cccnc2n1 C1(CNC(c2c(C)cc(F)cc2)=O)CC2CCC1N(C(=O)CCC1CC1(F)F)C2 c1(CC)cccc2[nH]c(C(N3CCN(C(=O)Cc4ccc(C)s4)C4CC34)=O)cc12 Cc1cc(=O)c(C(N2CCC(C)CC2)=O)cn1C1CC1.c1(N)ccc(F)c(F)c1 c1(C(N2CCCC(COC)(NC(=O)C(=O)N(C)C)C2)=O)cn2nccc2nc1C C1(C(=O)OC)CC(C)N1C(=O)CCCNC(C1(C)C=CCC1)=O c1(C(=O)NCCN(C(c2c(C)nc(C3CCOC3)s2)=O)C)sc(C#N)cc1Cl N1(C(CC(C)C)=O)CC(CCNC(c2c(Cl)nsc2Cl)=O)OC(C)C1 C1(CC)CN(C(=O)Cn2ncc(O)nc2=O)CCC1NC(C1CCNC1=O)=O N1(C(CC2CC(=O)OC2)=O)CCC(CF)(NC(=O)CCN2CCCS2(=O)=O)C1 CN1CC(C(=O)NCC2CCCC2NC(c2ccnn2C(F)F)=O)OCCC1=O c1(CC)cc(C)c(C(=O)NC2CN(C(c3ccc(NC(=O)NC)cc3)=O)CC2C)o1 C1(NC(C(C(C)C)NC=O)=O)CCN(C(=O)CC2(C)CCS(=O)(=O)N2)C(C)C1 Cc1nc(NC2CCCCN(C(=O)C3CCc4c[nH]nc43)C2)ncc1[N+](=O)[O-] Cn1nnc(C(N2CC(F)CC2CNC(=O)C=Cc2cncn2C)=O)c1C(F)F CCCCC(C(=O)N(C(C)C(N1CCCC1CCOCC)=O)C1CC1)NC(N)=O n1(C(C)(C)C)ncc(C(=O)NCCOC2CN(C(C3COC(=O)N3)=O)C2)c1Cl C(C1CCCN1C(=O)C=Cc1ccncn1)=CC(=O)NCCCCC=C c1(C(N(CCCNC(=O)CCC(C)SC)CC)=O)cnc2n1C(C)CCC2 C1(OC)Cc2ccccc2N(C(C2CN3CCN2CC3C)=O)C1 C12(C(=O)NC(c3[nH]nc(C(C)C)n3)C)COCC1CN(C(c1cnns1)=O)C2 C(=O)(CC(F)(F)C(F)F)N1CCC(CCOC)(NC(c2c(CCC)occ2)=O)C1 c1(OC)cc(NC(C)=O)cc(NC(C2CCN2C(=O)Cc2ccnn2C)=O)n1 c1(CC(C)C)ncc(C(=O)NCC2(NC(=O)CCc3ccncn3)CCOC2)s1 Cn1cc2cccc(C(N3CCC(NC(c4n[nH]cc4F)=O)C(O)C3)=O)c2n1 CCC(C)C(C(=O)N1CCC(C(C)NC(c2cc3n(n2)CCO3)=O)CC1)OC c1(C(=O)NCCNC(C2CN3CCN2CC3)=O)cnc(O)c2ncccc12 CC#CCCCC(=O)NCC(C1CCN(C(c2ccc(N)cc2C)=O)CC1)(C)O C1(CC(=O)NC(CCOC)CNC(=O)CCc2csc(C)n2)CCCC12CC2 c1(C(C(N2CC(COC)(CNC(=O)CCNC(C)=O)C2)=O)C)c(C)n[nH]c1C c1(C(=O)NC2C3CN(C(C(C)C4CC4)=O)C2C3)[nH]cc2c1CCCC2 c1(OC)cccc(O)c1OCC(=O)NCCCCC(C)NC(=O)CC1CSC1 C1(CCCC(=O)NC(CC#C)COC)CC=C(C)CC1 c1(N2CC(CC(C)NC(c3cnn(C)n3)=O)C2)nc2ccc(F)cc2o1 c1(C(=O)NCC2CN(C(C(C)N3CCC3)=O)C(C)C2)ccc2oc(O)nc2c1 c1(C(=O)NC2CN(C(c3cc(C)on3)=O)CC2F)cc(S(C)(=O)=O)ccc1F C(C)(C(=O)N1CCCC1)N(C(=O)C=CC1CCC1)CCOC Cn1cccc1C=C(F)C(N1CC2C(CNC(=O)CC3C=CCCC3)C2C1)=O c1(CC(=O)N(CC(C)NC(N2CCCCC2)=O)Cc2cccnc2)sc(O)nc1O C1(CNC(CCCc2nc(C)sc2)=O)CC2(CCN(C(c3cscn3)=O)CC2)C1 C1(NC(c2nc(C)[nH]c2C(F)(F)F)=O)CC2(C1)CC(NC(=O)C(C)C)C2 N1(CC(=O)NCC2(O)CC(NC(COCc3cc(C)on3)=O)C2)CCNC(=O)C1 CC(C(C)(C)C(=O)N1CCCC(C(N)=O)C1)NC(c1ncccc1Cl)=O Nc1c(C(=O)NC2CC(CNC(=O)CCOc3ccccc3)C2)cc(F)cc1Cl C1(C(C(=O)NCSc2ccccc2)N(CC(CC)(F)F)C)CCCC1S(C)(=O)=O C1(C(=O)NCCC2N(C(CC(C=C)(C)O)=O)CCSC2)CC2(C1)CC(C)(C)C2 C12(NC(c3c(C)cncn3)=O)CCC(CNC(=O)C(C)c3cc[nH]n3)(C1)OC2 C1(C(=O)NCC2OCCN(C(c3cccc(C#N)c3)=O)C2)CN2CCCCC2CO1 c1(CN2CCC(O)(CNC(C3CCC(C)CC3)=O)C2)cc2ccccc2[nH]1 C1(CN(C2CCN(C3CCOCC3)C2=O)C)CCCN(C(=O)CN2CC=CC2)C1 N1(C(c2c(C#N)cc(Br)cc2)=O)CCCC12CCN(C(C1CCCCO1)=O)CC2 C1(C(N2CC3C(CNC(C4CC(SC)C4)=O)C3C2)=O)Cc2ccccc2C1(C)C CN1CC(O)CC1(C)C(=O)Nc1cnc(Cl)cc1C(=O)O CC1=C(C(=O)NCC2CC(O)(CNC(=O)CC(F)(F)Cl)C2)SCCO1 N1(C(=O)C(c2ccc(Cl)cc2)C2CC2)CCN(C(c2cccnc2O)=O)C(CF)C1 C(C)(N=c1[nH]c(=NCCc2nccs2)[nH]c2cc[nH]c12)C1C(C)C1 c1(NC(c2scc(CNC(c3c(C(N)=O)cccc3)=O)c2)=O)c(Cl)cccc1Cl N1(C(C2C(=C)C2)=O)CC2CC(C1)C2NC(C1CC1C(F)(F)F)=O c1(C(N2CCC(OCC(=O)NCC3N(CCC)CCC3)C2)=O)cc(O)ccc1C Cc1cccc(C(=O)N(C)CC2CCCN2C(C2CC3(C2)CC(CO)C3)=O)c1F C1(CC(=O)NCC(C)N(C(c2cc(C(=O)OC)[nH]c2)=O)C)CC2(CCC2)C1 c12ccc(cc1F)Cc1cn(nn1)Cc1noc-2n1.C1(CCN)CCC1 C1(CCC(=O)N(C2CC3(CCC3)C2)C)CCN(C(C2(CO)CCCC2)=O)CC1 c1(SC)cc(NC(N2CCCCC2C(C)(C)O)=O)nn1C c1(C(C(=O)NCC2CC2)N(C(CC)C(=O)OC)C)cc2nc(Cl)ccc2o1 CC(C)C(O)CC(=O)N(C)CCNC(c1ccc(O)c(F)c1)=O c1(NC(CC2(C)CN(Cc3cc(Br)c[nH]3)C2)=O)nc(Cl)ccc1Cl c1(C(N)=O)cnc(Cl)[nH]c1=NCC1(NC(=O)C2=CS(=O)CCC2)CCCC1 C(C1OCCc2ccccc21)NCc1nc(-c2cn(C)nn2)sc1 C1(C(C)NC(C2CCCC2)=O)CCN(C(c2ccccc2C(C)(C)C)=O)CC1 N1(C(CC)(C)CNC(=O)N(C)CC2CCC(C)CC2)CCc2sccc2C1 c1(C(=O)NC2C(NC(CC3OCCC(C)(C)C3)=O)CC2)cnnc2ccccc12 N1(C(CC(COC)NC(C2C3CC(=O)CC23)=O)=O)CCC(CO)C(O)C1 C1(CC(=O)NCCCC(C)OC)CN(C(C2CC(C)C2)=O)CCO1 c1(C(=O)NC(C(C)NC(CC2CC(OCC)C2)=O)(C)C)cnn2ccn(C)c12 c1(C(=O)NCc2c(C(N(CC(O)C(C)(C)C)C)=O)con2)cnn(C)c(=O)c1 CCCCN=c1cc(NCCc2nc3ccccc3n2C(C)C)nc[nH]1 O=C1CCCCC(C(N2CCC(C(F)(F)F)C(CNC(C3(CF)CC3)=O)C2)=O)N1 C1(NC(c2c(OC)ncnc2OC)=O)C(C)CN(C(=O)C2=CCOC2)CC1C c1(C(=O)NCC2CC(NC(=O)CCc3cncnc3)C2)c(O)ccc(F)c1Br c1(C(=O)NCCOCCN(C)C(C2CCCC(=O)O2)=O)nc(=O)n(C)[nH]1 Cn1ccc(F)c1-c1ccc(C(=O)NC(C(=O)O)C2CCC2)cc1 CCCC(CNC(c1cnn(C2CCC2)c1)=O)NC(=O)CC1COCCO1.C1(C)CC1 C1(NC(C2N(C(C3C(C)N(C)CC3)=O)CC2C)=O)CN2CCC1(C)CC2 N1(C(c2c(C)cc(O)nc2)=O)CCN(C(=O)C(C)CC(C)(C)C)C2CCCC12 O=Cc1cccc(-c2ccccc2CNN2CCCCCC2C(F)(F)F)c1 C1(C(=O)NC2CCC(N(C(=O)Cc3csc(Cl)n3)C)CC2)CCn2nccc2C1 c1(CNC(CC2(C=C)CN(C(=O)C3=CCCCCCC3)C2)=O)ccccc1C(=C)C C12(CC)CCCN(C1)C2=O.c1(Nc2ccnc(C(C)(C)C)n2)cc(Cl)ncc1F Cc1nnn(CC(=O)N(CC(C)O)CCNC(c2cc(CO)[nH]n2)=O)n1 S(=O)(=O)(c1ccccc1F)N1CCC(CNC(C)C)C1.c12cc(c(Br)cn1)CO2 c1(OCC(=O)NC2CC(NC(CN(C)C(c3cccs3)=O)=O)C2)cc(Cl)cc(Cl)c1 C1(NC(CCn2ncc(C)c2)=O)CC2CCC(C1C)N2C(c1cn(C)cc1C)=O c1(OC)ccc2c(N3CCC(C#N)(NC(c4nccnc4Br)=O)C3)ncnc2c1 CCC(CC)CC(F)C(=O)NC(C1(O)CCN(C(=O)C=CCN(CC)CC)C1)C C1(NC(c2c(C)nc(C3CC3)[nH]2)=O)CC2CC1CN2C(=O)Cc1cccs1 CCC(C(=O)NCC(C)C(=O)Nc1cc(C)c(C)cc1C)C(C)(C)CC N12CCC(C3(CCC3)CNC(=O)CC(CC(C)C)CC1=O)CC2.CC(=O)OCC N1(C(C2C(C)CCO2)=O)CC=C(CC(=O)N2CC(C)(C)OC3(CCC3)C2)CC1 N1(C(C2(CCCC)CC2)=O)CCC(COC)(NC(c2csc(C)n2)=O)CC1 C1(N(C(C(N2CCN(C)CC2)C)=O)C)CCN(C(c2cc(Br)n[nH]2)=O)CC12CC2 c1(NC(C2CC=CCC2C(N2CCC(CC3CC3)C2)=O)=O)ccc(CO)nc1 N1(C(=O)Cn2cc(Cl)cn2)CCC2(CCCN2C(c2csc3ccccc23)=O)C1 N1(C(c2sccc2Cl)C(=O)Nc2ccc(F)cc2)CCC(OC(F)(F)F)CC1 c1(CCCOC(C2CC(SCN(C)C)C2)=O)c(F)cc(F)cc1F c1(-c2nc(C(=O)Nc3ccnnc3)sc2)cccc2c1CNC2=O C1(CC(=O)NCC23CC2CN(C(c2c[nH]ccc2=O)=O)C3)CC2C=CC1C2 C=CCC(CNC(=O)CC(C)SC)C(=O)NC(C)(CO)C1CCCC1 C1(CC(=O)NCCCCNC(=O)CCC2CCCO2)CC2(CCCC2)C1 c1(C(N2CCC(CO)C2C)C(=O)NC(C(=O)OC)C)cccc(CO)c1C C1(NC(CN(S(CC)(=O)=O)C)=O)CCCN(C(=O)C2=NNC(C(F)(F)F)C2)C1C CC1=NOC(=O)C1CCC(=O)NCC1CC(NC(=O)CCc2nc[nH]n2)C1 CC(C)CC(C)(O)C(=O)NC1CCCC(C(=O)NC2CC23CCOCC3)C1 c1(CC(=O)NCCCN(C(C2C(C(=O)OC)CC2)=O)C2CC2)c(C)noc1C Cc1cc(Cl)c(C(=O)NC2CC(NC(=O)CCc3nccn3C)C(O)C2)cc1F N1(C(C(=O)N(C)C)=O)CC(C(N2CCOCCC2CO)=O)CC(C(C)(C)C)C1 c1(CC)nnc(O)c(O)c1OCC.C12CC3(CC(C3)NCc3ccc(cc3)CN1)C2.C(C)CC c1(N2CC(C(N(C(c3c(F)cccc3F)C)C)=O)C2)ncnc2c1COC2 c1(C(=O)NCC=CCNC(=O)C2=CCOC2)ccc2nn[nH]c2n1 Cc1cc(C(=O)NC2CCC(CCNC(=O)CC(C)(C)C(F)F)C2)c(N)c(Cl)c1 C1(C(=O)NCCN(C(=O)CCCCN2C(=O)CCC2=O)CC)CC(S(C)(=O)=O)C1 c1(C(C)N(C(CN(C)CC2CC2)=O)C2CC2)nc(COC)cs1 c1(C(N2CCC(CC#C)(C(=O)Nc3ccsc3)C2)=O)n[nH]cc1[N+](=O)[O-] C1(NC(CCCOCC)=O)CCN(C(=O)C=CCOCC(F)(F)F)CCC1(F)F c1(OC)c(C)ccc(C(=O)N(C2CN(C(c3csc(Cl)n3)=O)C2)C)c1F C1(NC(C2C(C)C2)=O)CC2CCC(C1)N2C(c1ocnc1-c1ccccc1)=O C1(C)(C(=O)NCCOC(C)=O)CCN1C(=O)C(O)c1ccco1 N1(C(C=CC(=O)OCC)=O)CCC(CCNC(c2cc(CCO)on2)=O)CC1C C1(C(=O)NC2CC3(C(NC(C4(C(N(C)C)=O)CC4)=O)C3)C2)COCCC1(F)F C1(C(=O)OC)CCCCN1C(=O)CN(c1nccc(OC)n1)CCO C(C)(C(C)NC(=O)CNC(c1cscn1)=O)NC(C=C(C)Cl)=O N1(C(C(CC)(F)F)=O)CC2(CCCC(CNC(=O)CC(C)CC(C)(C)C)O2)C1 C(CC(CC)C(=O)N(C(CC(F)F)C(=O)NCc1cncn1CC)C)=CC CCC(C)CC(=O)N(C)CC1CCN(C(=O)CCNC(C2CCCCC2)=O)CC1 N1(C(C=C(C)C2CC2)=O)CCN(C(=O)CC2CCCOC2)C(CCO)C1 Cc1cc(C)c(CC(N2CC3C(CNC(=O)C=CC(=O)NC4CC4)C3C2)=O)s1 c1(NC2C(CNC(C3CCC(=O)N3)=O)CCCC2)ncc([N+](=O)[O-])cn1 N1(C(c2c(N)nccn2)=O)CC2(CC2)CC1CNC(=O)CCn1ccccc1=O CCCC(CC)CCC(=O)N(C(CC)C(=O)N1CC(C2CCN(C)C2)C1)C Cc1cc(NC(C2CC23CC(NC(=O)CCCCCF)C3)=O)cnc1F CCC(O)(C(=O)NCC(O)CNC(c1cc(OC)ncn1)=O)c1ccccc1 C1(C(=O)NC(C(=O)NCC2(O)CCCCC2)c2ccoc2)CCCCOC1 N1(C(c2c(C)nc(C(C)C)s2)=O)CCC(C)(CNC(=O)Cc2cccs2)CC1 CCC(CN=C(NCc1cccc(C2CC2)c1)NCC1CCCO1)CC(F)(F)F C1(CNC(CSCCN(C)C)=O)CCCCN1C(=O)C=Cc1cocn1 C1(C(N2CCC3(CC(NC(C4(C)CCC4)=O)C3)C2)=O)CC2COCC(C1)C2 c1(OCC)ccc(C(=O)NCCCOCCNC(C2C(C)C2C)=O)cc1N N1(C(=O)NCCCC=CC)CCCOC(c2ccccc2Cl)C1 C1(NC(C2(C(=O)NC)CC2)=O)CCN(C(=O)C(C)(C)C(C)C)CCC1CO C1(C(N(C2CCCCC2)CC)=O)CCN(C(c2ccc(I)c(O)c2)=O)CC1O Cc1ccc(F)nc1CNC(=O)N(C)CC=Cc1ccc(Br)cc1 c1(C(=O)NCC(CNC(CCc2cc(C)on2)=O)F)ccc(N)c(Br)n1 Cc1cccc(C(N2CCC(C)(CNC(C3CCC(=O)C3)=O)CC2)=O)c1C c1(NC(c2cn(CC)nn2)=O)ccc2ncnn2c1.C12CCC1C(=O)NC2 C1(CCC)CCC(O)(C(=O)N(C)CCn2cc(CC(C)(C)C(=O)O)nn2)CC1 C1(C(C(=O)NCCCOCCCNC(C2C(CC)C2)=O)C)CCCCCCC1 N1(C(C2C3(CC(NC(C4(CC)CCC4)=O)C3)C2)=O)CC2CCC(C1)C(=O)O2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(c2cc(C(=O)OC)sc2)=O)CC1C C=CCCC(F)(F)C(=O)NC1CCCCC1NC(C1CC(=O)NC(=O)C1)=O C=CCCCCCC(=O)NCC1(COC)CCN(C(=O)CC2CCCCO2)C1 Cc1nn(C)c(Cl)c1C=CC(N1CC(C)CN(C(=O)C(Cl)=CCl)C(C)C1)=O c1(C(=O)NC(C)CNC(=O)COCC2CC2)cccn2c(O)nnc12 C1(OCC(C)C)CCCN(c2nnc(CO)n2CCCCC2CCOCC2)C1 CCC(C(=O)NC(C1CCN(C(=O)C=CCF)CC1)C)C(C)O N1(CCn2cc(C(=O)OC)nn2)C(=O)NC2CC12CC(C)CSc1ccccc1 C(C)(C(=O)NCCCN(C(=O)Cc1ccco1)CC)OCC C12(NCC3(S(C)=O)CC3)CCC(C1)OC2 c1(C(NNC(=O)NC(C(C)C)CCOCc2ccccc2)=O)ccc(F)cc1F C1(N(C(Cn2c(C)nnn2)=O)CCF)CCCN(C(=O)C(c2ccc(F)cc2)O)C1 N1(C(=O)CC2CC23CC3)CC2(CCN(C(c3cn(C4CCCCC4)nn3)=O)C2)C1 N1(C(CCSCCC)=O)CCC2(CCC(NC(=O)Cn3ccc(C)n3)C2)C1 CCCCCCC(O)CCC(=O)Nc1cccc(NC(C2CCCC(=O)CC2)=O)c1 C(CC(O)C(=O)N1CC(O)(CNC(=O)C(C(C)C)N2CCCC2=O)C1)SC C1(NC(C=CC(CC)C)=O)CN(C(=O)CCCN2CCCC2)C(C)(C)C1 n1(CC(C)F)nc(-c2ccc(F)cc2)nc1Cc1sc(O)nc1O CC1CCN(C(C2CCCN(C(c3c(F)cccc3F)=O)CC2)=O)CCO1 c12ncc(c(C(F)F)n1)CN2.C1(C(=O)O)CSCCN1C(C1(C(F)(F)F)CC1)=O N1(C(C2C(CC)CCC2)=O)CCC(CNC(c2ocnc2C)=O)(OC)C1 C1(CNC(C2C(C)OCC2)=O)CC2(CC(NC(c3cnn(C)c3C(F)F)=O)C2)C1 N1(C(CC2CCC(NC(c3cc(CC)[nH]n3)=O)C2)=O)CCC2CCC(C1)N2C N1(Cc2scc(C(=O)O)c2)CCC(NC(c2cc(Cl)ccc2I)=O)C(F)C1 C1(CNC(C2CC(F)(F)CS2)=O)(CO)CCCN(C(C2CCCO2)=O)C1 c1(OC)cc(-c2ccncc2)ccc1CNCc1ncccc1OC C#Cc1cccc(C(=O)NCCC2(C)CCN(C(=O)C=CCO)C2)c1 C1(CNC(COCC)=O)CC2(CC2)CN1C(c1csc(C(F)F)n1)=O c1(C(N2CC(O)(CNC(=O)Cc3cccc(C4CC4)c3)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C12(NC(c3ccc(OC)c(F)c3)=O)CCCC1N(C(=O)Cc1nc(=N)[nH][nH]1)CC2 c1(CN2CCN(C(c3c(OC)c(Br)ccc3)=O)C3C2C3)ccc(C#N)cc1F N(C(=NCCN1CC(OC2CCOC2)C1)NNCCS(C)(=O)=O)CC(C)C#N CC(CCCCNC(c1cc(C#N)c[nH]1)=O)NC(c1cc(C(F)F)no1)=O C(=O)(C(C)(C)CCNC(=O)Cc1cnns1)NC1CCC(OC)C1 C(C1=NOC2CN(C(c3ccc(N)cc3F)=O)CC12)NC(C1(CCC)CCC1)=O Cc1cccc2c(C(=O)N(C(C)CNC(C3CCc4nccn4C3)=O)C)c[nH]c12 C12(C(=O)NC3CN(C(C)=O)C3)CC1CCN2C(c1cccc(-c2cnco2)c1)=O C(=O)(C1=C2CCCN=C2NN1)N(C)CC1(CNC(=O)C=C(C2CC2)C2CC2)CC1 C12(C(=O)NCCCC(C)NC(C3CC=CCC3)=O)CCCN(CC1)C2 c1(C(=O)NC2C(CNC(C3C(C)CN(C)C3)=O)CCC2)ccc(N)c(F)c1 c1(C(N2CCCC2c2c(F)cccc2F)C(=O)NCC2CC2)ccc(Cl)cc1Cl c1(N(C2CCN(C(CCC(=C)Cl)=O)CC2)C)snc(Cl)c1C#N C1(CNC(C(C)(C)c2cnco2)=O)COCCN(C(c2cccc(N)c2)=O)C1 Cc1nn(C)c(Cl)c1C(N1CCS(=O)(=O)CC1)C(=O)NCCCC1CC1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(CC(=C)C)C(=O)NC1COCCC1O C(=O)(CCCC(C)(C)C)NCC1C(C)CCCN1C(C1CCCO1)=O N1(C(CCC(=O)NCCC)=O)CC(NC(=O)Cn2ccnc2C)CC2(CC2)C1 CCC(CC(C)C)C(=O)NC(C1(O)CN(C(c2scnc2C(F)F)=O)C1)C c1(C(N2C(C(N3CCCCC(C)C3)=O)CC2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1Cl CC1(C)CN(C(c2nc(Cl)c(Cl)s2)=O)CCC1NC(c1ncc2ccccn12)=O c1(C(C)C(=O)NC(C)CN2CCN(C(=O)C3=CCC3)CC2)ccc(F)c(F)c1 Cc1cccc(C(=O)NC(C(=O)NC(C(C)C)c2cccs2)C2CC2)c1N N1(C(C(C)OCC=C)=O)CCCC(C)(CNC(c2sc(Cl)cc2Cl)=O)C1 c1(OC)cc(C)nc(N(C2CNCC2F)C(=O)Cn2nc(C)cc2C)n1 Cc1csc2ncc(C(=O)N(CC(C)CNC(c3onc4c3CCCC4)=O)C)n12 N#Cc1cccc(I)c1NC(C1CC(NC(c2c(F)cc(F)cc2F)=O)C1)=O c1(C(=O)NC(CC)CN(C(=O)CC2CCN(C)CC2)C)cc(N)nc(Cl)c1 C(=O)(CS(=O)(=O)C1CC1)NC(CNC(C1(C#C)CCCC1)=O)C(C)C C(C)(CN=c1[nH]c(=N)[nH]c(=NCc2c(Cl)cncc2Cl)[nH]1)NC(C)=O C1(NC(C(COCC)C)=O)CCCCCC1C(=O)NC(C)C(C)(C)O N1(C(C2(C#C)CCC2)=O)CC(NC(=O)CC2CCCNC2=O)C(n2ccnn2)C1 c1(CC(=O)NC(CN(C)C(C2CC2(C)C)=O)(C)C)cc(F)cc(F)c1 Cc1nc(N2C3CCCC2CN(C(=O)C2=CCS(=O)(=O)C2)C3)ncc1[N+](=O)[O-] n1(CC)nc(C(=O)N(C)CCNC(=O)CN2CCC(C)CC2)c(C)n1 C1(C(=O)NCCC(CC)(C)NC(=O)C(N2CCNC2=O)C)CNC(=O)CC1(C)C N(C(=NCCC(=O)NC)N1CCSC(C)(C)C1)CC(CC)C(F)(F)F Cc1cc(NC(=O)C(C2(O)CN(C(=O)COc3ccccc3F)C2)F)ccc1Br CC(C)(C(=O)N1CCC(OCCO)C1)C1=CCN(C(=O)Cn2cccnc2=O)C1 C1(NC(C(C(C)C)SC)=O)CC2CC1N(C(c1cncc(-n3ccnn3)c1)=O)C2 CCCC(C)CCCC(=O)N1CCOC(CNC(c2nccc3n[nH]cc23)=O)C1 C(=O)(CC1CCc2ccccc21)NCC1(F)CN(C(CC(CN(C)C)(C)C)=O)C1 CCC(C)(COC)C(=O)N(C1CCN(C(C2CC3C=CC2CC3)=O)CC1)C c1(NC(C23CN(C(c4cncc(CC)c4)=O)C(C2)C3)=O)cccc([N+](=O)[O-])c1 CC(=O)C(C)CCC(=O)Nc1csc(Cl)c1 C(=O)(C(F)C(C)(C)O)N1CC=CC(C(=O)NCC(COCC)C)C1 Nc1cc(C(=O)NC2CCC2C(=O)NC2(C3CCCCO3)CC2)cc(F)c1 C1(NC(=O)C(F)CC2CCCC2)(CNC(=O)COc2ccon2)CCCCCC1 C(=O)(C(F)C(C)(C)O)N(C(CNC(C(C)(C1CC1)OC)=O)C)C.c1(N)ccccc1F S(=O)(=O)(CC(=O)N1CC2CC1C2NC(c1cc(C(=O)OC)no1)=O)N(CC)CC Cc1c(Cl)ccnc1C(=O)N(C1CCN(C(c2sccc2C#N)=O)CC1)C C1(C(C)(C)O)(C(N(CC=C)CC)=O)CN(C(=O)COc2ccccc2)C1 c1(NC(=O)CSC(F)F)ccc(C(=O)OC)c(C)c1 C(=O)(CC(C)P(C)(C)=O)NCCC(C(C)C)NC(c1ccn(CCO)c(=O)c1)=O C(=O)(C(C1=CCSC1)N1CCC(c2cc[nH]n2)CC1)NCC Cc1cc(C)n2ccc(C(N3CCN(C(=O)C(=O)C(F)(F)F)CCC3C)=O)c2n1 C(C)(CCC(=O)N1CC(C)C1C(=O)N(C)CC1CCCO1)SC C1(NC(C2(COCC)CC2)=O)CCCN(C(c2cnc(S)n2C)=O)CC1 CC1(C)CN(C(=O)Cc2cncc(F)c2)C(CNC(c2ccc(O)cn2)=O)CO1 c1(OC)cc(C)ccc1C(=O)NCC1CC1NC(=O)CC(c1ccc(C)cc1)C C1(CCC)CCCC1C(=O)NCCn1cnc(C(N2CC(N3CSCC3=O)C2)=O)c1 c1(C(=O)NCCCC(C)NC(c2snc(O)c2Cl)=O)ccc2c(c1)CC(=O)N2 c1(C(C)C)cc(=NCCCSCCNC(C2(C)CC3CCC(C2)S3)=O)[nH]cn1 Nc1sc2c(c1C(=O)NCC1CCC(CO)O1)CCC2 CC1CN(C)CC(C(N2CC3CCCC3C2)=O)O1.c1(C2C(=O)N2)cccnc1 C1(CNC(C2N(CC)CC2)=O)CC(F)(F)CN1C(c1ccc(C(F)F)cc1F)=O CC1(C)CCC2(CC1)CN(CC(O)C(F)(F)F)C2 S(=O)(=O)(c1cc(Br)c(F)cc1F)NC1CC(C)CN(C(C2CCCCC2)=O)C1 C1(C(=O)OC)CCN(C(C2C3CN(C)CC23)=O)CC1(C)C c1(C(C(=O)NC(CCN(C(CC(C)n2ccnc2)=O)C)(C)C)C)ccccc1F CCC(F)C(=O)NCCNC(=O)C(C)OCc1ccc(Cl)s1 Cc1ncsc1CC(N1CC(OCCOC2CCCOC2)C1)=O.n12cc(nn1)CC2 c1(CC)cccc(CC)c1NC(=O)Nc1cccc(N(C)C(C)=O)c1F c1(NC(c2cc(-c3ccc(OC)cc3C)[nH]n2)=O)cc2c(C)cccc2[nH]1 C1(CN(C(C=COCC)=O)C)CN(C(=O)CCc2scnc2C)CCO1 C(C)(C)(C(=O)NCC(C)(C)NC(=O)COCC(=O)NC1CCOCC1)OC(C)C N1(C(c2c(OC)ccs2)=O)CC2CC(C(N3CC=CC3CF)=O)(C2)C1 c1(C(=O)OC(C)(C)C)ncc(C(=O)NCC(C2CC2)Sc2ncn(C)n2)s1 CCCC(CC)C(=O)NCC1CN(C(c2cnc(COC)s2)=O)C(C)(C)C1 c1(CNC2C3CN(C(C4(CCOC)CC4)=O)CC32)cc2ccccc2nc1C C(=O)(C(O)CCCNC(=O)CNC(=O)C(C)(C)C)NCCOC1(C)CCC1 C12(NC(c3ccnc(O)c3)=O)CCCC1N(C(=O)C=C1CCCC1)CC2 N1(C(c2cc(CF)on2)=O)CCCC(N2CCN(c3nnc(C4CC4)o3)CC2)C1 c1(CC)oc2ccccc2c1CC(=O)NC1CCCC1NC(C1(CC)CCC1)=O CC(C)C(C(=O)NCC#CC(=O)NC(C1CCCO1)C)NC=O C1(C(=O)NC2(C(=O)OC(C)(C)C)CCC2)OC2CCC1CC2 Cc1c(NC(c2csc(C(F)(F)F)c2)C)ncnc1N1CCC(C)C1 Cc1cnncc1C(=O)NC1CCOC(C(N2CC3C(CO)C3C2)=O)C1 C12(CCNC(=O)Cc3c[nH]ccc3=O)CCC1CN(C(C1(C(F)(F)F)CC1)=O)C2 Cc1cc(CC(N2CCCC(CCNC(c3cc(Cl)c[nH]3)=O)C2)=O)n(C)n1 c1(C(N2CC3C(CNC(C4C(C=C)OCC4)=O)(C3)C2)=O)ccc2c(c1)CCCN2 c1(C(=O)OCC)cc(C(=O)NC2CN(C(c3sccc3Cl)=O)C2)cs1 c1(C(=O)NCCCN(C(=O)C(O)C(F)F)CCC)ccc(=O)n(CC(N)=O)n1 CCCC(CC)C(=O)NC1CC(NC(C23CC(NC(=O)OC(C)(C)C)(CO2)C3)=O)C1 CCCC(C(=O)NC)NC(=O)NCC(=O)N(C(C)C(=O)NCC1CCC1)C C(CCCC(=O)NCC1CCCC1NC(C1CC(=C2CC2)C1)=O)OCCC=C Cc1cccc2ncc(C(=O)NCC3CC3NC(C3(CF)CC(F)(F)C3)=O)n12 C(=O)(CCCCCN(C(=O)CCN(C)C)C)NC(c1nc(=O)o[nH]1)C CC(=O)C(C)CC(C)C(=O)N1CCC(F)(F)C(CNC(=O)C=C(Cl)Cl)C1 c1(-c2n(C(C(=O)N(CCOC)C(C)C)C)ncc2)cn(C)nc1C(F)F C#CCCC(O)CCNC(=O)CSCCNC(c1coc(C)c1)=O c1(C(=O)NC(C(C)NC(CCn2c(C)ncc2)=O)C(C)C)c[nH]nc1S(N)(=O)=O c1(CN(CCOC)CC2CC3(CCC3)CO2)ccc2oc(O)nc2c1 N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(C2(C)CC(O)CN2C)=O)CC2(CC2)C1 C1(C)(C(=O)NCCOCCN(C)C)CC(NC(c2csc(-c3ccoc3)n2)=O)C1 N1(C(C2C(C(C)C)N(C(=O)CNC=O)CC2)=O)CC(N2CCCC2)C2(CC2)C1 C(=O)(C(C)(C)C(C)C)OCc1ccc(C)cn1 c1(C(C)(C)C)csc(C(=O)NC2CCC(CNC(=O)CSC(F)(F)F)C2)c1 C1(CNC(C)=O)CCN(C(=O)Nc2ccnc(-c3ccoc3)ccccc2)C12CC2 c1(C(N2C3C(NC(Cc4cc(OC)ncc4)=O)C(C3)C2)=O)c(C)ncn1OC N1(C(C2(OC)CCN(C(c3nc(CC)sc3)=O)C2)=O)CC(=O)N(C)C(C)C1 N1(C(C(c2ccc(C)cc2)CN)=O)CCS(=O)(=O)C2(CCCCC2)C1 N1(C(C2CCC(n3cc(-c4c(C)cccc4)nn3)C2)=O)C2CCC1CC1(CC1)C2 Cn1ncc(Br)c1CN1CC2C(CNC(C3COCCO3)=O)C2C1 c1(N2CCC(NC(C)=O)CC2)nc2c(c(=NCC3OCCC3C)[nH]1)CCC2 C12(C(=O)NOCCOCCO)CC(CN1C(=O)CC1CNC(=O)O1)C2 C1(C(=O)NCC2(CN(C(=O)C(F)(F)c3ccccc3)C)CC2)CCC12CCC2 N1(C(COC(CC)C)=O)CCC(CC(N2CC(CN=[N+]=[N-])C2)=O)C1 CC(C)C(CCC(=O)NCSc1cccnc1)NC(C)C(F)(F)F c1(C(=O)NC(C(C)(C)NC(C(CSC)O)=O)C)c(C(F)F)nc2n1CCCC2 Cc1cc2[nH]c(C(N3CCC(NC(=O)CC4CCCC(C)(C)O4)C3C)=O)cc2s1 c1(C(N2CCCC(C)(COC)C2)=O)cc2cc(Br)ccc2s1 CCCCC(CNC(C1(F)CC1C)=O)NC(=O)C(=O)Nc1ncc[nH]1 c1(CCC)n[nH]c(=NC2CCC3CN(C(c4ccc(F)c(CO)c4)=O)CC3C2)s1 C(=O)(C(C)(F)C(C)(C)F)N1CCC(c2cn(-c3cccc(Cl)c3OC)nn2)(NC)C1 c1(OC)ccc(C(=O)NC2CCC(NC(c3cc(C#N)c[nH]3)=O)C2)c(N)c1F c1(OC)ccc(Br)c(CNC2CCCN(C(C3CC3(F)F)=O)C2)c1F C(C(C)(O)C(=O)NCC1CCC(CNC(=O)CCNC(=O)C(C)(C)C)CC1)OC CC1=C(C(=O)N2CC=CC2C(N2C3CCC2CC3)=O)CCO1 N1(C(c2c(C)cno2)=O)CC(CNC(=O)C(C)OCCN(C)C)C(O)C1 N1(C(C(C(CC)C)O)=O)CCCC(C2(NC(=O)Cn3ccc([N+](=O)[O-])n3)CC2)C1 c1(OC)ncc(Cl)c(C(=O)NC2(C(=O)OC(C)(C)C)COC2)n1 C(=O)(CC(CC)C(C)C)N(CCCNC(=O)C(O)CN(C)C)CCOC c1(C(=O)NCC2C(NC(c3cc(C4CC4)no3)=O)CCC2)nc[nH]c2nccc1-2 CC1CN(C(c2ccc(CF)cc2)=O)CC1NC(=O)CCC1CCCCO1 c1(C(=O)NC(CC)CN(C(=O)CC2CCC(C(F)(F)F)O2)C)cc(C)cc(N)c1 C1(NC(c2c(CCC)n[nH]c2)=O)CC2CC(NC(C3(C(N)=O)CC3)=O)CC12 N1(C(C(CC)(C)CO)=O)CCC(C2CC2)(CNC(=O)Cc2cccc(C)c2F)C1 c1(CNC2C(C(=O)Nc3nc(C)nc(O)c3)CCC2)ncc(Cl)cc1[N+](=O)[O-] N1(C(c2cn(CCC)nc2)=O)CCC(CCF)(NC(C2CCN(C)CC2)=O)C1 c1(C(=O)NCCN(C(c2cncc(Cl)c2)=O)CC2CC2)nccc2[nH]ccc12 CCCC(CC)C(=O)N(C(C(=O)NCC1CCN(C)CC1)C1CC1)C Cc1cc(C(=O)NCCC(C)N(C)C(c2cccc(C(=O)N(C)C)c2)=O)sc1C N1(C(C(C(CC)O)C)=O)CCc2ccccc2C(N(C)C(=O)C=CBr)C1 n1(CC)cnc2c(NCCc3cncn3C)[nH]c(=NC(C)c3ccsc3)nc12 C1(NC(COCCCCCC)=O)CCCCN(C(c2cc(C#N)cs2)=O)C1 CC1CC(O)CCN(C(c2cccc(C(=O)NCC3CCCC4(CC4)C3)n2)=O)C1 c1(NC2CC(NC(c3ccc(F)cc3Cl)=O)C2)ncnc2cc(Br)ccc12 C(CC(=O)N(Cc1ccc(C)o1)OC)C1CCN(C(C2C(C(=C)C)OCC2)=O)C1 CCC1=C(C(=O)N2CC(O)(C(C)NC(C3CC4CC3C3CC43)=O)C2)CCCO1 C1(CN(C)C)CCC(N=c2[nH]c(N(C)Cc3c(C)cccc3Cl)nc(=N)[nH]2)CC1 C1(CC=C)(NC(C2CC2C(F)F)=O)CN(C(=O)C(C)OCCOCC)C1 CCC(C(=O)NC1CN(C(c2cc(NS(C)(=O)=O)co2)=O)C1)c1cccnc1 CC1(C)C=C(C(=O)N2CCOC(CCCNC(C3CC3Cl)=O)C2)C1 c1(NC(c2cc(NC(C3C(C(=O)OC)C3)=O)c(C)cc2)=O)c(F)cc(F)cc1Cl C#CCCC1=C(C(=O)OC)C(c2cnn[nH]2)NC(=S)N1c1ccc2c(c1)OCO2 C1(c2n(CCCCCC)nnn2)(N(CC(=O)OCCCC)C(C)C)CCN(C)C1C c1(C(N2CC(CNC(C3CCC4C3C4(F)F)=O)C2)=O)cc2cccn2c(O)n1 C1(NC(CSCCCC)=O)CC2CCC1CC2NC(=O)C=Cc1cnc(C)s1 C1(CNC(c2c(C)sc(O)n2)=O)COCCN(C(=O)CC2(C)CC2(F)F)C1 c1(C(=O)NC2C(NC(C(CC)Nc3ccccc3)=O)COC2)ccc(C)c(C)n1 CCC(C)(C)CC(=O)N(C1CCCC1)CCNC(=O)C(CCOC)OC c1(N(C)CCF)nc(=NCC23CCCN2CCC3)[nH]c2c1SCC2 CCCCC(CC)NC(=O)C(NCP(C)(C)=O)=O C1(C)(CC)CCC(C(=O)NC(C2CN(C(=O)C(O)C3CCCC3)CCO2)C)O1 N1(C(COc2ccc(CC)cc2)=O)CCC(NC(=O)CSNBr)C(O)C1.C1(O)CCCC1 C1(NC(C(CCCNC(CCOC)=O)O)=O)CC2CC1CC21CC1 C1(C(N(CCN(C(c2ccsn2)=O)CC)CC)=O)CCC12CCCO2 [N-]=[N+]=NC1CC2CCC1(NC(C1(Nc3ccccc3)CC1)=O)C2 N1(C(c2c(C)ccnc2)=O)CC2(C1)SCCC2NC(C1CCCC(C)C1)=O N1(C(C2C(C(C)C)C2)=O)CCOCC(C(=O)NC2CC(O)C2O)C1 N1(C(Cc2cccc(OC)c2)=O)CC2(CC(CC(N3CCC(CF)CC3)=O)C2)C1 C(CCCCC(=O)N1C(C(=O)N(CC(O)CO)CC)CC2CC12)=CC C1(NC(CCc2cnc(C)s2)=O)C2CN(CCNC(=O)CNC(=O)N(C)C)CC12 c1(C(=O)NC(CN(C(C(c2ccc(C)o2)C)=O)C)C)cc2n(n1)CC(C)(C)CO2 CN1CC2CCC1C(NC(c1ccc(CNC(C3CCCC34CCC4)=O)o1)=O)C2 c1(OCC(N2CC(NC(c3n(CC#C)ccc3)=O)C2)=O)cc(C)cc(C)c1 c1(C(N2CC(NC(C(CC)N(C)C)=O)C(OC)C2)=O)ccc(C)c(Br)c1N C1(C(=O)NCC2CCCOC2)CC2CN(C(c3c(F)cccc3Cl)=O)CC2C1 CC1CCCCN1CCC(=O)OCC1CC(COc2ccccc2C(=O)O)C1 CC(C)CC(O)CC(=O)N1CC2CC2(CNC(=O)CCC2CC2(Cl)Cl)C1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC2CCC1N2C(=O)C=Cc1cccn1C N1(C(C(COC(C)C)(C)C)=O)CCC2C(C(N3CC(SC(F)F)C3)=O)C2C1 C1(OC)CC2(C1)CC(C(N1CCC(O)(CN(C)C(C3CNC(=O)N3C)=O)C1)=O)C2 c1(OC2(C(F)(F)F)CC(COC)N(S(C)(=O)=O)C2)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 N1(CC)CCN(C(C2CCCN2C(C2CCCC2OC)=O)=O)CC1=O Cc1ccc(C(N2CCCCC(NC(=O)C(C)(C)c3nncn3C)C2)=O)c(C)n1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CCC(C)(NC(=O)CCc2cn(C)cn2)C1 N1(C(c2nc(COCC)sc2)=O)CCN(C(C2CCC2(C)C)=O)C(CC)C1 c1(C(=O)NC2CC(NC(C3OCC4CCCC34)=O)C2)ccnc2c1CCC2 C#Cc1ccc(NC(C2CCC2NC(c2occc2C(C)C)=O)=O)cn1 c1(OC)ccc(N)c(C(=O)NCCCCC(CO)NC(=O)C=CC2CC2)c1 C1(CNC(c2ccc(C)cc2)=O)CCCCCN1C(c1cnc(C)[nH]1)=O c1(C(=O)NCC(C)N(C(CN2CC(CC)C2)=O)C)cncc(C)c1C N1(C(C2CN(C(c3ccc(C(C)C)o3)=O)CC2(C)C)=O)CC2(CCC(=O)N2)C1 C1(C(=O)NC2(COC)CN(C(C3CCCC(F)C3)=O)C2)C2CC3C(C2=O)C13 C1(CNC(C=CCN(C(=O)Cn2cnnn2)C)=O)CNC(=O)N1 c1(OC)cccc(Cl)c1C(=O)NC1CN(C(c2ccccc2CO)=O)CC1C Cc1c(Br)sc(C(=O)NCCNC(=O)CCc2ncc[nH]2)c1Br C(=O)(C(CCOC1CCCC1)CCO)N(CC(C)O)C.C1(=O)CO1 C1(NC(C(C)S(N)(=O)=O)=O)CCCC(N=c2nnn(C)[nH]2)C1 c12cccnc1N(CC)CCCNC(=O)C2.c1(C(=O)NC)cc(Br)cs1 C1(CN(C(=O)COC(F)F)C)CN(C(C2CCS(=O)(=O)N2)=O)CCO1 C(CCC(=O)O)N(C1(CCOC(=O)COC(C)(C)C)CC1)C.C(C)(C)(C)NC(N)=O CC(C)CC(C)C(=O)NC1CC2CC1N(C(c1ccn(-c3cccnc3)n1)=O)C2 C(C(C)(CNC(c1nnnn1C1CCCC1)CC1CCCOCC1)CO)OC CC1Cc2c[nH]nc2C(C(=O)N2CCN(Cc3cc(F)c(Cl)cc3Cl)CC2)C1 CN1CCOC(C(N2CCCC2C(=O)NCCCSC(F)F)=O)C1 c1(-c2occ(-c3nc(CC(CC)C)nn3C(C)C(C)(C)C)n2)c(F)cccc1Cl N1(C(C(c2ccccn2)C)=O)CCCCC1C(C)Nc1cc(F)ncn1 c1(C(=O)NCC(C)(CO)NC(c2c(C)ncn2C)=O)ccc(C)c2ccccc12 O=C(C#CC1CCCOC1)NC1CC1NC(c1cnc2n(c1=O)CCS2)=O C#CCC(C)(C(=O)NCC1(n2ccnn2)CC1)NC(C1(C#N)CCCO1)=O C(=O)(CCCCCCCC)NC(CCN(C(c1cncc(C=C)c1)=O)C)C Cc1nc(C(N2CCC(CN(C)C(C3C(F)(F)C34CCC4)=O)C2)=O)cc(O)n1 c1(CC(=O)NCC2C(NC(C3(COC)CC3)=O)C2)cc(Br)cc(Br)c1 Cc1cn(C)cc1C(=O)NC(CC1CCOCC1)C(=O)NOCCCC1CC1 N1(C(c2n(C)cc(Cl)c2)=O)CCC(O)CC1C(N1CC=CC1)=O N1(C(COCCC=C)=O)CC(C)(C(N2CCC(CCCC)C2)=O)C1 C(=O)(C1=C(Cl)CCOC1)NCC1CCC(NC(c2ccc(Br)cc2F)=O)C1 N1(C(C=CC(=O)OCC)=O)CC2CCC1CN2C(C1CCN(C(C)=O)C1)=O CCCC(C(=O)NC1CC(C(=O)NC(C23CCC(CO2)C3)C)C1)NC(N)=O CCC(CC(F)(F)F)NC(C1CCN1C(=O)CC1CSC1)=O CC(C(=O)NCCCC1CN(C(c2cnsn2)=O)CCO1)S(N)(=O)=O c1(C(N2CCN(C(=O)C=Cc3ccoc3)C(CF)C2)=O)cc2n(n1)CCCC2O N1(C(C=CCOCCOC)=O)CCC(C)(CNC(c2nnn(C)n2)=O)C1 C1(C(N2CC3C(NC(c4cccc(C)c4Cl)=O)C3C2)=O)CC(=O)NC2CCCCC12 C1(C(=O)OC(C)(C)C)CCCOC1(C)C.c12nc(cs1)CC(=O)N2CC#C Cc1ccc(-c2ocnc2C(=O)NC2CCC2CNC(C2CC3(CC3)C2)=O)cc1 C1(C)(CNC(C(C)C)=O)CCCN(C(c2ccncc2-c2ccccc2)=O)C1 c1(NC(=O)NC2CC3CCC2N3)cc(C2CCOCC2)ccc1F C1(C(=O)NCCCCNC(C(C)N(CC#N)C)=O)CC12C(=O)Nc1ccccc12 CCC(C)(COC(CO)C(C)C)C(=O)NCc1nc(C)ccc1F c1(OC)ccc(C(=O)NCC(C)(C2CC2)NC(c2cc(F)c[nH]2)=O)c(N)c1F c1(C(=O)NCC(CCCC)NC(C2CC(F)(F)C2)=O)ccc2nccc(C)c2c1 c1(C(=O)NC(CC)CNC(C2(C)CCC(=O)N2)=O)cc([N+](=O)[O-])nn1C C1(N)CCN(c2ccc(-c3cccc(C(=O)O)c3)cc2)CC1F.OC(F)F CC(C(=O)NCc1coc(C2CC2)n1)S(C)(=O)=O N1(C(C(C(=O)OC)CC)=O)CCC2CN(C(=O)CCCN(C)C(C)C)CC2C1 N1(C(C(C2(C)CC2)NC(c2ccccc2)=O)=O)CCC(C(=O)CO)CC1 c1(C(N2CC(N(C)Cc3cc(Cl)cc(Cl)c3Cl)C2)=O)cc(Cl)c(Cl)cc1F c1(CC)c[nH]nc1C(=O)NCCCCNC(C12CC(CC(C)C)(C1)C2)=O C=C(C)C(C)(C)C(=O)NCC1CC(C)N(C(=O)CCNC(C2CCC2)=O)C1 Cn1ccc(S(=O)(=O)N(C2CCN(C(c3ccc(Cl)cc3)=O)CC2)CCO)n1 c1(CC(N2CC(OC)(CNC(C3CC3C(C)(F)F)=O)C2)=O)c(C)nn(C)c1C c1(C(N2CC(C)(NC(CCn3c(C)nc(C)n3)=O)C2)=O)c[nH]c2c(Br)cccc12 N#Cc1ccc(C(N2CC(NC(c3cc(Br)nc(Br)c3)=O)C2)=O)c(F)c1F Cc1cc(C(=O)NC(C)(C)CNC(C2CCSC(C)C2)=O)c2cccnc2c1C C(=O)(CCCCN(C)C(=O)CC(C)(C)C#N)NC(c1n(C)cnn1)CO c1(C(=O)OCC)c[nH]cc1CC1CC1.C1CCCN(C)C(=O)C(=O)N1 CN1CCCC1CCC(=O)NC1CCN(C(=O)Cn2ccc(C3CC3)n2)C1 C(C)(CCC(=O)N1C(CNC(c2cc(C(N)=O)co2)=O)CC2CC12)OC C=CCC(C)(C)CC(=O)N1CCCC(N(c2cc(C(=O)OC)nc(Cl)n2)C)C1 Cn1ncc(S(N)(=O)=O)c1C(=O)NC1CCC1NC(c1cccc2c1OCO2)=O C=C(Cl)CC(C(=O)NC1CCCCC1CCO)NC(=O)CC(C)(F)F c1(CC(=O)NCC=CCNC(c2[nH]cc3c2CCC3)=O)cc(O)nnc1O c1(C(N2C(C)CCC(NC(c3c(C)ncs3)=O)C2)=O)cc(F)c2[nH]nnc2c1 O=C(C1CCCn2ccnc21)NC1CC2(C1)CN(C(=O)CC(C(F)F)C1CC1)C2 C1(O)(CNC(C(CSCC)NC(=O)CCC2CC2(F)F)=O)CCOCC1 C(=O)(C(C(C)NC(=O)C(CO)C(F)(F)F)C(C)C)NCC1CC(CC)C1 N1(C(c2nc(CNC(C3CC(C(C)C)C3)=O)oc2)=O)CCOCC(O)C1 c1(OC)ccc(CC(=O)NCC23CC2CN(C(=O)C(C)(C)F)C3)c(Cl)c1 c1(C(N)=O)ccc(C(=O)NNC(=O)N2CCCCC2)cc1Cl Cc1ccc(N(C)CC2(C)CN(C(=O)NCc3ccccc3)C2)o1 c1(C(N2CCC(NC(C=C(CC)C)=O)(CF)C2)=O)ccc(C)cc1Br C1(NC(C2N(CC)CCC2)=O)CCC(C)(CNC(C2(OC)CCC2)=O)CC1 N1(C(C(C)N(C(C)=O)C)=O)CCC(F)(C(=O)N(C2CC2)Cc2nncn2C)C1 C1(CC(N2CCCC(N(C(C(C)C)=O)CCO)C2)=O)CCC2(CCC2)CO1 C1(CNC(C(C)(C)SC)=O)CCC(NS(C)(=O)=O)CC1 c1(C(=O)NCC2(CN(C(=O)CCCOC(C)(C)C)C)CC2)cc[nH]c2nccc1-2 N1(c2ccnc(NCCN(C)CCO)n2)CCCC(C2CC2(F)F)C1 CCC(O)C(C)C(=O)NCC1CCN(C(=O)Cc2ccc(O)c(O)c2)C1(C)C Cc1nnccc1C(=O)NCC1CC1NC(c1ccc(C(C)(F)F)cn1)=O N1(C(C2N(C)CCC2)=O)CCSCC1CCNC(=O)CC1(n2ccnc2)CC1 N1(C(C2(CC=C)CC2)=O)CCCC2(CNC(=O)CCc3ccc(O)nn3)CC12 C1(NC(c2ccccc2Cl)C(=O)NCCCOC)CC(OC)C1(C)C C1(NC(C(C(=O)OC)OC)=O)CCCCCN(C(=O)C=C2CN3CCC2CC3)C1 N1(C(C2(C=C)CC2)=O)CC(CCNC(c2csc(CC(F)(F)F)n2)=O)OC(C)C1 N1(CC(=O)NCC2N(C(C3N(CCC)CCC3)=O)CC2)CCC(O)CC1 CC12CCOC(CNC(=O)C(C)(C)CNC(C3C4CCC(F)C34)=O)(C1)C2 N1(C(C(CCSC)OC)=O)CC2(CCC2)CCC1CNC(C1CC(F)(CF)C1)=O c1(NC(CC)=O)ccc2[nH]cc(CC(=O)NNC(=O)c3c(Br)noc3C)c2c1 c1(C(=O)NCCC2(NC(=O)C=CCF)CC2)[nH]nc2ncc(Br)cc12 C(CCCC(=O)N1CCC(C(=O)NC(CC(N)=O)C2CC2)C1C)N(C)C CCCCC(C)CCC(=O)NC1CCCC1NC(=O)C(=O)N=S(C)(C)=O O=C(CCS(=O)(=O)C1CCCC1)NCC1CCN(C(=O)C(F)CC2CCCC2)C1 N1(C(=O)CC2CCC2)CCCC(C2CCN(c3ncc4ccsc4n3)CC2)C1 c1(C(=O)NC(CC)(C)C)ccc(CNC(=O)CC(C)SC)nc1 C1(CNC(=O)C2=CSCS2)CN(C(c2ccnn2C2CC2)=O)CCCO1 c1(C(N(C(C)Cc2cccc(C)c2)CC)=O)ccc(OC)c(C)c1 c1(NC(=O)CSC)cc(F)c(F)c(F)c1.CCC1(c2ccccc2)CN1 C1(n2cc(CNC(c3ccc(COC)s3)=O)nn2)CCCC1(C)O C=CCC(C)C(=O)N1CCC(C)(CNC(=O)CC2(CS(C)(=O)=O)CC2)C1 N1(C(CC(CC)C2CC2)=O)CC2(C)CC1(C(=O)Nc1ccc[n+]([O-])c1)C2 Oc1cc(CNC2CCOC(CSc3ccccc3)C2)ncn1 c1(CC)cc(F)c(C(=O)N(CCCNC(=O)C(C)C2CCOC2)C)cc1F CN1CCOC(C(N2CC(NC(c3ccc(C#N)o3)=O)C(n3ccnn3)C2)=O)C1 N1(C(CN(CC)CC2CCCC2)=O)CC(C(c2ccc(C(N)=O)o2)=O)OC(C)C1 Cc1sccc1C(N1CC(O)(c2cn(CC=CCSC3CCCO3)nn2)C1)=O c1(OCC(=O)NC(C)C(C)NC(c2cnn(C)c2Cl)=O)ccc(S(C)(=O)=O)cc1 Cc1cnn(CCCC(=O)NCC2(C(N)=O)CN(C(c3scnc3C(C)C)=O)C2)c1 C1(C(N2CCC(C)(NC(c3[nH]c(=NC)sc3)=O)C2)=O)CCc2nc(O)[nH]c2C1 C=C1CC2(C1)CC(C(=O)NCCCN1CCN(C(=O)C(O)C3CC3)CC1)C2 c1(C(CO)NC(C=CC(=O)OCC)C)cccc(C)c1 c1(C(C2CC2)NC(C2(CNC(C3C(C)(C(C)CC)C3)=O)CC2)=O)c(C)cnn1C C(=O)(CC(CC)C(F)F)N(CCC(=O)NCCCCC(C)C)CCCC C1(OCC)CCCC(CC(=O)NCC2CC2NC(=O)CC2CCCC2(F)F)C1 N1(C(C2CCCN(C(CCCC3C(C)C3)=O)C2)=O)CC2C=CC1CC2 CC(C)CCCC(C)C(=O)NC(CCN(C)C)C(=O)NCC1(C)CCCC(=O)N1 CC1(C)OC2(C(N3CCCC(CNC(=O)C(F)(F)CO)C3)=O)CCC1CC2 CC1CCCC(C)N1CCC(=O)NCC1(CNC(C2CCCC2)=O)CC1(F)F Cc1ncc(C(N2CCCC(C)(NC(c3cc(O)n(C)n3)=O)C2)=O)cc1C#N C1(CNC(C2CN(C(C)C)C2)=O)CCN(C(=O)CCCCO)CC1C c1(C(N(C(C(=O)NCc2ncnn2C)c2cccs2)C)=O)ccc(CO)nc1 N1(C(C(C)CN(C)C)=O)CCCC(CC(=O)NCc2ccsn2)CC1 C(=O)(CC1=CCN(C(=O)COCC2CC2)CC1)NC(COC)C(C)C c1(OC)c(C)cc(C(=O)NC(C)C(CO)NC(c2[nH]nnc2C)=O)cc1Cl CCCCC(C(=O)N1CCC(OCC(C)C)C1)NC(C1CCNC(=O)C1)=O C1(NC(=O)C2=CCN(C(=O)C=C(C3CC3)C3CC3)C2)CCc2nn[nH]c2C1 C=C=C(C)CC(=O)NC1CC(NC(c2ccc(N3CCCC3)cc2)=O)C1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(C2CC23CCSCC3)=O)CC1F C=CCC(CNC(=O)COCCOCCOC)NC(=O)CCCC1CC1C CN1CCCCC1CCC(N1CCCC(NC(c2ccncn2)=O)C1)=O C1(N(C(C2C(CCC)C2)=O)C)CCCN(C(=O)C(F)(F)C2CCOCC2)CC1 CC1(C)CN(C(=O)CC2CCCNC(=O)C2)C(CNC(=O)C2=CCSC2)CO1 c1(CNC(COCC)=O)cncc(C(N2CCCC(CCO)C2)=O)c1 c12ccc(c(C(F)(F)F)c1)c(=O)[nH]2.c1(NC(C2(CC)CC2)=O)cc(O)ncc1C C=CC(C)(C)CCCNC(C1(CNC(C2CCC(C)(C)CC2)=O)CC2(CC2)C1)=O N1(C(C2CC3CCC3C2)=O)CC2CNCC2C1.c1(C(C)(C)C)cc(C=O)no1 c1(CNC(C2CCCN(Cc3ccc(C(=O)OC)nn3)C2)=O)ccc(F)cc1Cl C(=O)(CCN1C(=O)COc2ccccc21)N1CC(NC(=O)C2=CCC2)C(F)C1 N1(C(C(C)CO)=O)CC2=C(C1)CN(C(c1cc(Br)ccc1Cl)=O)C2 N1(CCC(CC)C2CNC2)CCN(C(=O)Cc2ccccc2)CC1 c1(C(N2CC(CC)(NC(=O)CC3CCCC34CC4)C2)=O)ncc(C)cc1F c1(C(=O)NC2CC2CNC(=O)C(Cc2ccccc2)C2CC2)ncccc1Cl N1(C(CNC(CC)=O)=O)CCN(C(=O)Cc2ccccn2)C2(CCC2)C1 N1(C(C(C(C)C)NC(=O)CC2CCC2)=O)CCN(C)CC(C)C1 C(C1c2ccccc2CCN1C(=O)CCC(=O)c1ccccc1)NC(CCC#C)=O c1(C(=O)NC2CN(C(C3CN(C(C)=O)C3)=O)C2)c(C)nc(C)n1O c1(C(N2CCCC(N(C(CCC)=O)CC)CC2)=O)nc2cccnc2s1 C(c1cccc(OCCOC)c1)=CC(=O)NCC1(C)CCC(NC(CCC)=O)C1 N1(C(C(C=C)C)=O)CCC(C(C)NC(=O)CCCn2cc(F)cn2)CC1 N1(C(C(COC)(F)F)=O)CCc2sccc2C1CNC(=O)C(C)OCCC(C)C C(CCCC(=O)NCCCN(C(=O)C(=O)C(C)C)C)N(C(C)C)C N1(C(=O)CN2CCCNC2=O)CCCC(F)(CNC(C2C3CCC2CC3)=O)C1 c1(OC)ccc(C=CC(N2CCC(C)CC2CNC(=O)Cc2ccoc2)=O)nc1 c1(C(N2C(C(C)NC(=O)C=Cc3ccsc3)CCC2)=O)cnn(C)c1N C1(C(C(=O)NCCCN(C2CCCCC2)CCC)OC(C)=O)CC=CCC1 C1(C(=O)NCC2CCN2CCCCc2nccs2)(COC)CCC1 C12(CCCCC1)NC(=O)c1cn(nn1)C1(C)CCN(C1)C(=O)CC2.C1(OC)CC1 c1(CNC(C2CC(OCC)CC2O)=O)cc2c(C(F)(F)F)cccc2s1 C(=O)(C(O)CCCNC(c1cccnc1S)=O)N1CC(CS(C)=O)C1 C1(CC)CC(C(=O)NC(C)(C)CN(C)C(c2ccnc(OC(C)C)c2)=O)CCO1 CC1CN(C(C2CCC(C)O2)=O)CC(C(N2CCOC(C(N)=O)C2)=O)O1 c1(C(=O)NCCC(C)NC(C(CCCC)=O)=O)cc(Br)c(C)cc1C C1(C(=O)NC(C=CC(N2C(C)(C(=O)OC)CC2)=O)C)CC2C(C1)C2(F)F C1(NC(C(c2ccccc2)NC(C2C(C)C2)=O)=O)C2COCC12 C(CC(C)C(=O)NC1COCCC1C(=O)NCC(=O)NO)OC c1(CC)c(Br)c(C(N2CCN(Cc3ccc(I)c(F)c3)CC2CC#N)=O)nn1C N1(C(=O)NCC)CCCN(C(C(=O)CN2CCOCC2)=O)CC1.CN c1(CCO)cnc(Sc2nnc(N(C(CN(C)C)(C)C)C)o2)nc1O C=CCCCCCC(=O)NCC1CN(C(=O)CSC(F)(F)F)C1 c1(C(=O)NCCCC(C)NC(=O)C(F)CC2CC2)cccnc1O C1(NC(CCOCCCOC)=O)CC2CN(C(c3cscn3)=O)CC12 CC(C)(C(=O)NCC1CCCC1NC(C1CC12CC2)=O)c1ccno1 C1(CCCC)CN(C(=O)CCCNC(C)=O)CCN1C(=O)C(C1CC1)OCC Cc1nnc2n1CCCC2C(=O)NC1CCCC1NC(c1ncc(F)cc1F)=O N1(C(C2CCC(CC)O2)=O)CCC(CNC(C2CCCCC2)=O)C(C)C1 C1(NC(c2cn(CC)nc2)=O)CCCCC1NC(c1c[nH]nc1-n1cnnn1)=O c1(C(N2CC(NC(C3CC4C=CC3O4)=O)C2)=O)ccc(C2CC2)cc1F c1(C(N2CCCC(C(=O)NCC(=O)NCC)C2C)=O)cc(OC)cc2c1OCC2 C1(C2N(C(C3CC(O)(CC#C)C3)=O)CCC2)CCN(C(c2coc(O)n2)=O)CC1 N1(C(C(CC(F)F)NC(CCOCC(C)C)=O)=O)CCC2CCCC2CC1 N1(C(c2ccc(CNC(=O)C(F)F)o2)=O)CCC(O)C12CCC2 c1(-n2cc(CN(CC(=O)O)C(C3(C)CC3(Cl)Cl)=O)nn2)cccc2c[nH]nc12 C1(NC(C(C)(C)c2cccs2)=O)CC(O)CN(C(c2occc2F)=O)C1 C=CC(CC)C(=O)NCC(C)(O)CNC(c1csc(COC)n1)=O C1(NC(CNC(C2(C)CCC(=O)N2)=O)=O)CCn2ncnc2C1 c1(C(=O)NCC2(O)CN(C(CC(C(C)C)(F)F)=O)C2)cc2c(Cl)cccn2n1 Cc1cccc(C(N2CCN(C(=O)C(c3ccc(Br)cc3)C)CC2)=O)c1C C1(CC(=O)NCC2CCCN2C(=O)C(c2c(C)n[nH]c2C)C)(OC)CCOCC1 CC1C(NC(=O)C(F)F)CCCN1C(c1ccc(C(c2ccccc2)=O)[nH]1)=O C1(NC(CCCN(C(C)=O)C)=O)CC2CCC1N2C(=O)Cc1nc(C)sc1C [N-]=[N+]=NCCC(=O)NCc1occc1C(=O)NCCCC1CCCCO1 N1(C(C2CC(CCC)OCC2)=O)CC2CC(NC(=O)Cn3cc(C)cn3)C2C1 C1(NC(c2scc(C)c2Cl)=O)CC2CC(C1)N(C(=O)C(C)OCC(C)C)C2 N1(C(C(C2CCOCC2)C)=O)CCCC1CC(=O)NCC(C)OC(F)F C(=O)(C(CC)C(C)C)N(CC(C)C)CCOC.C(C)(=O)OC N1(C(C(C=C)O)=O)C(C(=O)NCc2cccc(C)c2)CC2CCCC12 CCCC(CNC(c1ccc(C)c(C)c1)=O)C(=O)NCC(C)(O)C(C)CC CC1=CCC(C(=O)NC(C)CCN(C)C(C2C3CCC2CC3)=O)CC1 c1(CN2CCCC(CNC(C3CC3C3CC3)=O)C2)ccc2cc[nH]c2n1 N1(C(Cc2c(OCC)nccc2)=O)CCCC(CC)(NC(C2CCC2(C)C)=O)C1 N1(C(c2nccc(N)c2Cl)=O)CCC2(CC1)CN(C(C1CCCC3(CC3)C1)=O)C2 N1(CC(=O)NCC(CCNC(COCC(=O)OC)=O)O)Cc2ccccc2C1 c1(C(=O)OC)cnc(NC(c2ccccc2)CC2CCOC2)cn1 N1(C(c2c(C)cc[nH]2)=O)CCC2(CCN(Cc3cc(Cl)sc3Cl)C2)C1 C(=O)(CCCCC1CC1)NCC1CC(CNC(=O)CCn2ccnn2)OC1 N1(C(=O)NCc2cc(OC)ncc2Cl)CC(C(F)(F)F)CC(C)C1 C1(C(=O)NCC2(CNC(CCOCC(C)C)=O)CC2)CCC2(CCCO2)CC1 C(CCC(C(=O)NCCCN(C)C(C)=O)NC(c1cccnc1S)=O)OC CC1CN(C(=O)C(C)(C)C2CCCCO2)CC(C)N(C(=O)CC2CC(F)(F)C2)C1 S(=O)(=O)(c1ccc(N2CCC(C(C)C)CC2)cc1Br)N(CC(CC)O)CC1CC1 c1(C(=O)NCC(CNC(c2c(CC)non2)=O)(C)C)cc(F)c(F)c(Cl)c1F N1(C(c2cn[nH]c2)=O)CC2COCC2(C(N2CCCCC2c2ccccc2)=O)C1 c1(C(=O)N(C2(C(=O)NCC(C3CCC3)C3CC3)CCC2)C2CC2)cc(F)c[nH]1 c1(NC(=O)NCC(CC)Oc2cccc(C)c2)ccc(-n2cccn2)cc1C CC1OCCCC1C(=O)N(O)Cc1cn(C2CCOCC2)nn1 C1(CNC(C(C(=C)C)(C)C)=O)CCN(C(C2CC2COC)=O)C12CCC2 c1(CC(N2CC(C#N)N(C(c3ccccc3)=O)CC2)=O)c[nH]c2ccc(Br)cc12 C(=O)(C(C)(C)C1=CCN(C(=O)CN2CCCC2)C1)N1C(C)COCC1 C(=O)(CCCN=[N+]=[N-])NC1CC(CNC(C2CC(CC)C2)=O)C1 N1(C(C2CC(O)(CC#C)C2)=O)CC2CCCC2C12CC2.C12CC(C1)CC(=O)N2 N1(C(C2CCN(C)C(=O)C2)=O)CCC(F)(F)C(CNC(c2cc(O)nn2C)=O)C1 c1(N2CC(C)C(C)C2)ncnc2c1ncn2CC(O)CN1CCCC1 c12cc(Cl)ccc1NC(=O)C2(F)F.C(C)(C(C)OC)C1(C)C(C(=O)OCC)C1 Cc1ccccc1CN(C)CCn1cnc(C(=O)O)n1 N1(c2n(-c3ccc(C)cc3)nnn2)CCN(C(=O)CC2CC(F)(F)C2)C(C#N)C1 C1(CN(c2ncncc2I)C)CCCN(C(c2csc(Cl)c2)=O)C1 C1(O)(CC(=O)NC2(C3CCCN3C(c3cncs3)=O)CC2)CCCC1 c1(N(C(CC)=O)CCC2CCCNC2)cc(N(c2ccon2)C)nc(C)n1 c1(C(N(CCCN(C(CC2CCC(C)C2)=O)C)C)=O)cccc2c1ccn2C C1(C)(C(=O)NCC(C=C)O)CCCN1C(=O)CCCCSC c1(CC)cc(F)ccc1C(=O)NC(C)(CNC(C1CCCN1N=O)=O)C1CC1 C12(C(N(C3CCN(C(c4cc(CO)n(C)n4)=O)C3)C)=O)CC3CC1C2C3 N1(C(c2cnn(CC)c2C)=O)CCCC(O)(CNC(=O)CCC2CC2(Cl)Cl)C1 c1(N(CCC)CCNC(C2(C)CCCCNC2=O)=O)nc2ncc(Cl)cc2o1 c1(C(N2CC(C3OCCN(C(C=C(COC)C)=O)C3)C2)=O)cccc(C(N)=O)n1 C(=O)(C(F)C(=O)NC(c1ccccc1)CNC(=O)CC1CCCOCC1)OCC c1(C(=O)NC(C2CCN(C(=O)C3CC3)C2)C)cc2cccc(Cl)c2[nH]1 C(=O)(C1=CCC(C)CC1)NC(C1(O)CN(C(c2ccc3n[nH]cc3n2)=O)C1)C C(C(F)(F)C(F)(F)F)n1c(-c2nc(C)[nH]n2)nnc1C(C1CCOC1)N C1(C(=O)NCCC2(OC)CN(C(C3CC(O)C(F)C3)=O)C2)CCC(N=[N+]=[N-])CC1 O(N=C1CCCCCC1)CC(=O)NCC(C)N(C)C(c1csc(Br)n1)=O C1(NC(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CCCSC2CC2)CC1O Cc1cc(C(C)(C)C(=O)NCC2CCN(C(C3C4CCCCC34)=O)C2)ccc1F c1(CNC(CCC=C)=O)ccc(N2CCN(C(=O)CC3CN(C)C3)CC2)cc1 C1(C)(C(=O)NC2CCC(NC(CCNC(COC)=O)=O)C2)CNC(=O)C1 c1(C(N2CC(CCNC(CCCC=C)=O)OCC2)=O)ccc(Cl)c(Cl)c1O Cc1ccc(Cl)c(OCC(=O)NC2CCC(CNC(C3(C)CC3(F)F)=O)CC2)c1 CC1NCCC1CNC(=O)Nc1cn(C)cn1 CC1(C)COC(CCNC(=O)CC(C2CC2)NC(=O)Cn2cc(C#N)cn2)C1 O=C1COc2ccc(S(=O)(=O)N3CCCCC34CCOCC4)cc2N1 c1(CC)cc(CC(=O)NCC2CC(NC(C3CC(N(C)C)C3)=O)C2(C)C)n(C)n1 CN(CCCC(=O)N1CC2CC1C2NC(=O)CC1CC(=O)NC1=O)N=O c1(C(=O)NC2C=CC(CNC(C3CC3(F)F)=O)C2)cccc(Cl)c1 C1(C(CNC(C2(CN(C)C)CC2)=O)NC(CSCC(C)C)=O)CCCC1 c1(CC)ccc(NC(C2(NC(=O)CC3(OCC)CC3)CC(F)C2)=O)c(F)c1 C(C(COC)CC(=O)N(C)CCN(C(=O)CC(C)CN(C)C)C)OC CCC(C)(C)C(O)C(=O)NC1CCCC1NC(c1ccccc1CC(=O)OC)=O CCC(CCC(=O)NC1CC(=O)N(C)C1)NC(c1cnnc(O)c1)=O c1(CC(C(N2C(CNC(c3n(C)ccn3)=O)CCC2)=O)O)ccccc1Cl N1(C(C(C)(C)O)=O)CCOCC2(C1)CN(C(c1ccc(F)cc1F)=O)CCCO2 C(=O)(C1CCc2c[nH]nc21)NCC=CCNC(C1CCC(C2CC2)C1)=O C(=O)(C(O)CCC(C)C)NC1CC(NC(c2cnnc(C)c2C)=O)C(O)C1 C1(CNC(C(CC2CCCC2)NC(C2CN(C)C2)=O)=O)OCC2CCC1C2 N1(C(C=Cc2c(C)nccc2)=O)CCC(NC(=O)C=CC(C)C)CC(C)(C)C1 c1(C2N(C(C(c3nc(C(N)=O)cs3)C)=O)CC2)cn(CCN2CCCC2)nn1 N1(C(CC(N2CC(NC(N)=O)C2)=O)=O)CC2CCC(C1)O2 C1(NC(CC2N(CC)CCC2)=O)CCN(C(c2cnns2)=O)CC1 N1(C(C2C(NCc3c(C(=O)OC)cccc3)C=C2)=O)CCC(O)C(O)C1 N#Cc1ccc2c(C(N3CC4C(C3)N4C(=O)CN3CCOC3=O)=O)c[nH]c2c1 CC(C)C1C(=O)NCCO1.C1(=CC(=O)NC2CN(C(=O)C3CC3)C2)CCCCC1 C1(OCC)CC2CN(C(=O)CN(CC(C)(C)NC(=O)Cc3ccoc3)CC)CC12 c1(C(=O)NCC2CN(C(C(C(=C)Cl)(C)C)=O)CC2(C)C)ccc2c(c1)CCOC2 C1(C(=O)NCC2N(C(C3OCCN(C)C3)=O)CCCC2)CCC(C)(C)CC1 C(=O)(C(C)(C)CC(=O)NC(CCOC)C(=O)NC(CO)CCOC)OCC C12(NC(c3ccc(OC(F)F)cn3)=O)CCN(C(c3ccsc3)=O)CC1C2 N(C(=NCCC)NCC(C1CCOCC1)(C)C)C(C#C)CCC c1(C(N2CC(CCNC(C(CC)C)=O)OCC2)=O)sc2[nH]c(C)nc(=O)c2c1C C1(C)(C(=O)NC2C(C)CN(C(c3ncc(F)cn3)=O)C2)CCNC(=O)C1 N1(C(CC(C)O)=O)CCN(C(c2ccc(C3CC3)cc2F)=O)CC1CC(F)(F)F N1(C(Cc2cccc(OC)c2)=O)CCCC2(CCCN2C(c2cccn2C)=O)C1 CCC(CC(F)(F)F)C(=O)N1CCC(CO)(NC(=O)Cc2cc(C)ccc2O)C1 CC(O)CCCCCC(=O)N1CCN(C(=O)CCS(C)(=O)=O)C(c2ncc[nH]2)C1 C(CC(=O)N(CC(C)(C)COC)C)(CC(C)C)NC(c1cc(CC)on1)=O c1(C(=O)NC2CCN(C(C(C)OCC)=O)CC2F)cc2ccccc2nc1O N1(C(C2ON=C(C)C2C)=O)CCC(O)C(N(C(=O)Cn2ncc(Cl)c2C)C)C1 N1(C(C2COCC(C)(C)O2)=O)CCC2(CCCN2C(=O)CC2CCOCC2)C1 c1(C(=O)OC)cncn1CC(=O)NCCNC(=O)CC1COC(=O)N1 c1(OCCOC)ccc(C(=O)NC2CC(NCc3csc(CO)n3)C2)cc1 CN1N=C(CC(=O)N2CCCCC2CCNC(c2c(F)cncc2F)=O)CC1=O Cc1cc(CNC(=O)CC2CCC(NC(=O)CC3CC(F)(F)C3)C2)n(C)n1 C1(C2(NC(C3CCN(c4ccc(Br)cc4)C3)=O)CC2)(OC)CCC1 C1(C(N2CCCC(CN(C)C(C3CCCCO3)=O)C2)=O)CCCCC1(F)F N1(C(C(C2(OC)CCCC2)(F)F)=O)CC2(COC(CNC(=O)C(C)N(C)C)C2)C1 c1(C(N(CC(C)CNC(c2cc(C(N)=O)c[nH]2)=O)C)=O)[nH]cnc1C#N C(=O)(N1CCCCCO1)NCCC(CCC=C(C)C)C C1(C(=O)NCC2CN(C(Cc3scc(C)c3)=O)C(C)C2)CC(=O)CC12CCC2 Cc1n[nH]c2cnc(C(=O)NC(CO)C(C)NC(C3(CN(C)C)CCC3)=O)cc12 c1(OC)ccc(OCC(N2CC(CNC(c3cc(C)c(C)s3)=O)C3CC23)=O)cc1 n1(CC)cnnc1C(=O)NC(C)CCCNC(C1(CC(F)(F)F)CCC1)=O C(=O)(C(C)(C)CNC(c1cscc1Cl)=O)NC(C)Cc1nc[nH]n1 c1(C(=O)NCC(C)(C)NC(c2ccc(C3CCC3)cc2)=O)cc(N)nc(Br)c1 Cn1ncc(C(=O)NC2(CCCNC(=O)CC3CC(F)C3)CC2)c1S(N)(=O)=O N1(C(C2CCN(C)C2)=O)CC(NC(c2cccnc2O)=O)CC(C)(C)C1 c1(OC)cccc(C(=O)NCCN(C2CCCCC2)C(C2CCC(F)(F)C2)=O)c1N N1(CC(=O)NC2(C)CC(NC(c3ccc(CC#N)cc3)=O)C2)CCS(=O)CC1 c1(C(=O)NCC2C3CN(C(c4n(CC)cnc4)=O)CC32)ccnc2c1ncn2C n1(CCCC(=O)NC2CC(F)(CNC(C3C(C)CCC3)=O)C2)cnc(C#N)n1 C(S(=O)(=O)c1cc2cc(F)ccc2s1)C1C(C)(C)C(N)CC1 c1(-c2c(OC)cc(F)c(C)c2)cnn2cc(C(N3CC4(C3)CC4(F)F)=O)cnc12 c1(C(N2C3CCN(C(c4cccn4C4CC4)=O)C3CC2)=O)cc2ncccn2n1 C1(C(=O)NC(CNC(C=CCCC)=O)(C)Cn2cccn2)Cc2ccccc2O1 C1(NC(C(C=C)CC)=O)CN(C(c2cc(OC)ccn2)=O)CCC12CCC2 c1(Cn2c(Sc3ccccc3)nnc2)ccc(CCC(C)CN2CCCC2)cc1 C1(N(CC(=O)Nc2cc(F)ccc2Br)C(C)C)COC2(CCNCC2)C1 c1(CC(=O)NCC2N(C(C(C#C)(C)C)=O)CCCC2)ccc(OC(F)F)c(F)c1 c1(NCC(CNC(c2c(C(C)C)n[nH]c2)=O)O)cc(O)nc(O)n1 N1(C(C(CC=C)c2ccccc2)=O)CCNCC12CCOCC2 c1(CNC(CC(=O)OC)CN)cc(F)c(OCCC(C)C)c(F)c1 C(=O)(CCCCCCOC(=O)NC1CCCCC1)NC(c1ncc[nH]1)CC c1(C(=O)NCC(CNC(c2cc(CC(C)C)nn2C)=O)OC)cncc(Cl)c1C CCCCC(CC)C(=O)NC1C2CC1N(C(c1ccnn1CC)=O)C2C O=S(=O)(c1csc(-c2ccc(F)cc2)n1)N1CCN(C2CCSC2)CC1 C(CCCCN1CCCC1)(C(=O)O)NC(c1c(CCC)n(CC)nn1)=O C1(NC(CSCCCC)=O)CCC2(CC1)CC(NC(=O)C(C#N)C(C)C)C2 C(=O)(C(C)(C)C(C)(F)F)NCCN(C)C(c1ccn(-c2ccccc2Cl)n1)=O c1(C(=O)NCC(CC)NC(C2(CSC)CC2)=O)cnc2nc(Cl)ccc2c1 C(CNC(c1cnn(CCO)c1N)=O)(C(C)(C)C)NC(c1cn(CC)nc1)=O C(C(CC(=O)N1CCCC1CCO)C1CCC1)NC(c1c(C)csc1)=O C1(NC(C=CC=CC)=O)CCN(C(=O)C(C)(C)CN2CCCOCC2)CC1CC C1(NC(CNC(C(CC)C)=O)=O)CC(F)CN(C(=O)C=CCN2CCOCC2)C1 C=CCCCCCC(=O)N1C(C(=O)NCCC(C)(C)F)CCC12CC2 Cc1cccc(C(=O)NC2CCC2CNC(C2CC2c2ccc(F)cc2)=O)c1F N1(C(c2ccncc2F)C(=O)NC)CCN(C(C)=O)C(C)C1 c1(OCC)ccc(N(CCCNC(=O)Cc2ccccc2)C)cc1OC c1(NC(=O)NCC(CC(=O)OC)(C)C)cc2c(cc1[N+](=O)[O-])OCO2 N1(CC(N2CCOCC2Cc2cccc(Cl)c2)=O)CCc2ccccc21 CC(C)(CNC(=O)COCCF)CC(=O)NCC1(O)CCOC1 N1(C(C(CC)(C)F)=O)CCN(C)C(CNC(=O)C(c2ccc(F)cc2F)(C)C)C1 O=C(CC1COCc2ccccc21)NNC(=O)c1ccc(C2CC2)o1 CC(CC(C)C(F)F)NC(=O)CC1CCN1C(c1sccc1CO)=O N1(Cc2c(C)n(C)nc2)CCC2(CC1)CN(C(=O)C(C)N1CCC1)CCO2 C(CNC(C1CCCC1CN=[N+]=[N-])=O)(CCNC(=O)CCSC)OC C1(NC(c2c(CC)non2)=O)CC2CN(C(C3CCCCNC3=O)=O)CC12 n1(C(C(=O)N(CCC(=O)NCCNC(C2(S)CC2)=O)CC)C)ccc(C)c1.CO c1(N(CC(C)C)C)ccc(C(=O)NC2CC(C)(NC(C3CCC(C)O3)=O)C2)cn1 Cc1cc(C)c(C(=O)NCC2CCCN(c3ncc[nH]c3=O)C2)s1 C1(CNC(C2(CC)CCOCC2)=O)CCCCC1NC(C1CCSC1)=O Cc1[nH]nc(C(=O)NCC2(CC(N3CC4(CSC4)C3)=O)CC2)c1Cl N1(C(C2(OC)CCC2)=O)CC2CC(NC(c3c(C4CC4)cnn3C)=O)CC1C2 C1(C(=O)NC(C)CCCNC(=O)Cn2ncnn2)C2CCC1CC2 N1(C(CC(CC)(F)F)=O)CC2CC1CCN2C(=O)CSCCC(F)(F)F N1(C(C2(CNC(Cc3cn(CC)nc3)=O)COC2)=O)CC(C)N(C)CC1C C=C(C)CCC(=O)NCC(O)CNC(=O)Cn1nc(C)cc1C(F)F C1(CC=C)(C(=O)NCc2cc(C)ns2)CN(C(=O)CC2(N(C)C)CC2)C1 CCC(C)CCCC(=O)NC(C)C(C)C(=O)N1CCOCC1 C1(CNC(C(c2c(C)noc2C)C)=O)CN(C(=O)Cc2cncnc2)CCCO1 c1(NC23C(NC(C(C)C4CC4)=O)CC(CC2)C3)c(C#N)cnc2ccc(Cl)cc12 C(=O)(C1CC(=O)Nc2ncn(C)c21)NCC1(O)CCCN(C(C2CC(C)C2)=O)C1 N#Cc1ccccc1-n1nc(C(F)(F)F)cc1NC(C1(n2cccn2)CCC1)=O c1(C(=O)NC(C(C)NC(CN2CC(CC)C2)=O)C)cn(C)nc1C(C)(C)C C1(CNC(c2cccc(=S)n2O)=O)CN(C(=O)Cc2nc(O)n[nH]2)CC12CCC2 C(C)(C)(CC(F)C(=O)NCC(O)(CO)CO)NC(c1c(C)c(O)ccc1)=O C(CCCCC(=O)NCCOCCC(=O)N(CC(C)CO)C)N.CCO CCC(C)CCCC(=O)N(CCC(=O)N(CC(C)(C)C#N)C)C C1(C(C)C)CN(C(=O)CN2CCSCCC2)CCN1C(C1CCC(=O)N1)=O N1(C(c2c(C)n(C)nn2)=O)CCOCC(C(=O)NCc2ncn(C3CC3)n2)C1 c1(C(N(C2CCCC2)CCNC(=O)CN2CC3CC3C2)=O)ccn(CCO)c(=O)c1 N1(C(c2cc(C)cc(C)c2)=O)CCC(C2CC2)C1C(=O)NCCP(C)(C)=O c1(CC(=O)N(CCNC(Cc2nnc(C)o2)=O)C(C)C)cn2cccc(C)c2n1 CC1CN(C(c2cnc(O)n2C)=O)CC1(C)CNC(c1cccc(CC#N)c1)=O N1(C(CCC=C(C)C)=O)Cc2n[nH]cc2C1C(=O)NC(c1cnn(C)c1C)C C#Cc1cccc(C(N2CC(C(=O)NC(C)(CC)CCO)(COC)C2)=O)c1C N1(C(C(C2CCC2)OC)=O)CC2CC1C2NC(=O)CC(C)(C)C1CCC1 c1(NCC2(C)CCCC2)ccc(-c2nc(C(c3ccccc3)(F)F)no2)cc1F N1(C(Cc2ccc(OC)cc2)=O)CCCC2(NC(=O)C=CC(C)(C)C)CC2C1 c1(C(N(CCC#N)CCSC2CCCO2)=O)nc(C(F)F)cs1 c1(C(N(CC(C)NC(=O)C(C2CCOCC2)C)C)=O)c(Cl)ccc2c1OCO2 c1(OC)cc(CNc2ccnc(C(=O)Nc3cn(C)cn3)c2)cnc1OC c1(NC(=O)N(CCC2CCCCO2)C2CC2)ccccc1Cn1cccc1 c1(COC(C(C)(C)C)=O)cccc(CNc2ccccc2)c1 Cc1cccc(CS(=O)C(C)C)c1F CC(C)CC(F)C(=O)NC1CC2(C1)CC(NC(c1sccc1-n1ccnn1)=O)C2 c1(CC(C(N2CC(C#C)(F)C2)=O)F)ccc(OC(=O)NC)c(F)c1 C1(NC(COCc2onc(CC)n2)=O)CN(C(c2ccncc2C)=O)C2CC12 N1(C(C(C)NS(C)(=O)=O)=O)CC(C(N)=O)(CNC(C2CC(F)C2)=O)C1 C1(NC(c2c(C(C)(C)C)c[nH]c2)=O)CC2CC1CN(C(c1cc(Cl)c[nH]1)=O)C2 c1(C(N(CCCN(C)C(C2CCC(=O)N2C2CC2)=O)C)=O)cc(N)ccc1Br c1(CC)cccc(CC(=O)NC(C)CC(C)CC)c1 c1(OC)ccc(CNC(=O)CNC(=O)CCCC(=O)c2ccc(F)cc2)cc1C N1(C(C(CC(=C)C)NC(=O)CCOCC2CC2)=O)Cc2cccc(F)c2C1 N1(C(C=C(CCC)C)=O)CCCC(C)(C)C1C(=O)NC1CC(=O)N(OC)C1 C1(c2nc(COC(C)C)on2)CN(C(c2cncc(F)c2Cl)=O)CCN1C.N1CC1 c1(CC(N2C(CNC(c3ccc(CSC)o3)=O)CCC2)=O)nn(C)cc1Cl C12(C(N3CC(C(C)(C)C)C3)=O)CCC(CC1NC(=O)CCN=[N+]=[N-])C2 N1(C(c2cncc(NCC)c2)=O)CC(NC(c2cccc(=O)o2)=O)C(C2CC2)C1 C12(C(c3nn[nH]n3)NC(c3ccco3)=O)CCCC1NCC2 C1(CNC(c2nn[nH]c2Cl)=O)CN(C(c2cnn(C3CCCC3)c2)=O)CC12CC2 N1(C(c2nc(C(=O)OC)cs2)=O)CC(F)(F)CC1C(=O)Nc1ncc(F)cc1O S(=O)(=O)(C1CN(C(C2C=CCCC2)=O)C1)N1CCN(C(=O)Cc2cc[nH]n2)CC1 C1(F)(CNC(C2CCCC2(F)F)=O)CCN(C(c2nn(C(F)F)cc2Cl)=O)C1 c1(C(=O)NCc2c(C(N(C(C)COC)CC=C)=O)con2)cn(C)cc1C C(=O)(C(C(CC)CC)OC)NCC1COCCN(C(C(C2CCC2)OCC)=O)C1 C1(CN(C(C2CCC(C)C2)=O)C)C2CN(C(c3ccsc3Cl)=O)CC12 C(=O)(C(C)(COC)CC)N1CCC(CNCC(=C)CC)C1c1ccco1 Cc1cccc(C(=O)NCC2(C)CCCN2C(c2ccc(C(N)=O)o2)=O)c1Br Cc1cc(C(F)F)oc1C(=O)NCC1(NC(=O)C=Cc2cccn2C)CCCC1 N1(C(C=CCCC)=O)CC(CNC(c2c[nH]nc2-c2cccs2)=O)C2CC12 c1(C(=O)NCC(C)(C(C)C)NC(C=CCCC=C(C)C)=O)cc(O)cc(C#N)c1 C(=O)(C(C)(C)CCNC(=O)C(C)CC#N)NCC(C)OC Cc1ccc2c(n1)N(C(=O)C=O)CCC2.c1(CC)ccccc1 Cc1cc(CNC(=O)CC=CCNC(C2CN(C)CCO2)=O)c(C)s1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CC2(CO)CC1(C(N1CC3CC3C3CC13)=O)C2 C1(NC(C2C(c3n(C)ccc3)C2)=O)C2CC3CN(C(=O)COC(F)F)C1C3C2 c1(OC(C)C)ccc(Br)cc1C(N1CCC(C(=O)NCc2nccs2)C(O)C1)=O C(C(=O)N=c1ccn(CC(N)=O)[nH]1)(C1CCCO1)NC(c1ccc(C#C)cn1)=O C1(SCCNC(CSC)=O)CCC(C)(NC(C2COC(C)C2)=O)CC1 Cc1csc(C=CC(=O)NCC(C)CNC(=O)Cc2occc2C)n1 c1(C(N(CCN(C(=O)CC2CCOC(C)(C)C2)C)C)=O)ccc2nnc(S)n2c1 N1(C(C(C)NC(C)(C)C)=O)C2CCC1CN(C(C1(C3CC3)CC1)=O)CC2 c1(CN(CCNC(COCC(=O)NF)=O)C(C2CCCS2)=O)ccccc1 Cc1ccc(C(=O)NCCCCC(C)NC(=O)CCOC2CCOC2)c(F)c1Cl C1(NC(CN(C)C(N)=O)=O)CS(=O)(=O)CC1[N+](C(=O)C(F)(F)C(F)F)(c1ccsc1)[O-] C1(CNC(C2ON=C(C)C2)=O)CC(NC(=O)C=Cc2ccsc2)CCO1 CC(C)CC(C)CC(=O)NCC#CCNC(c1cc(C(F)F)on1)=O C1(NC(Cc2cc(C)cc(C)c2)=O)CN(C(C2CCOC2C)=O)CC(C)(C)C1 C(=O)(C(C(C)(C)C)SCC)NCC(CC)NC(=O)CNS(=O)(=O)C1CC1.C(C)(=O)N c1(CC(C)C(=O)NC(CO)C(C)NC(=O)CC23CCC(CC2)C3)ccc(F)cc1 CC1CC=CCC1C(N1CCC1CC(=O)NC(C1CCCC1)CO)=O C1(NC(=O)CNC(N2CCCC2)=O)CC12CCC(NC(=O)Cc1cn[nH]c1)CC2 N1(CC(N2C(C)CC(NC(=O)CC3CCCC(C)C3)C2)=O)C(=O)NC(C)(C)C1=O c1(C(=O)NC23CC(NC(C4N(CC)CC4)=O)(C2)C3)ccc(C(C)OC)nc1C C1(N(C(COCCCCC)=O)CC2CC2)CCN(C(c2ns[nH]c2=O)=O)C1 C(=O)(CC(C)(C)CNC(C1COCCC1C)=O)N(CCOCC=C)C C(=O)(C1=CCCCC1)N(C1CCCC1)CCNC(C(C)(N(C)C)C1CC1)=O c1(COC(C2CN(C(=O)OC)CCN2Cc2ccccc2)=O)ncc(Br)cc1F CCC(C)C(C(=O)NCCCOCC(C)C)N(C)C(c1csc(Cl)c1)=O N1(C(c2nc(-c3cn(C)nc3)sc2)=O)CCC2(CCN(C(=O)C(C)(C)F)C2)C1 c1(CCCN(C(C(c2cn(C)nn2)N(C(=O)OCC)C)=O)CC)cc(C)cc(Br)c1 Cc1c2ccn1CCNC2=O.C1(C(=O)OC(C)C)CCC2CC12 c1(C(=O)NC2(C)CN(C(CC3CC(OC)C34CCC4)=O)C2)cccn2cncc12 N1(C(C2(C=C)CCC2)=O)CC(NC(=O)Cc2cc(COC)on2)C(C)C1 C(=O)(C1=CC(C)CC1)N(CCC)CCNC(c1ccc(SC(F)(F)F)o1)=O N1(C(CCOC(C)=O)=O)CCCN(C(=O)C(C)Cc2cccnc2)CC1CO C1(S(C)(=O)=O)(C(N2C(CCC)CN(C(=O)Cc3ccns3)CC2)=O)CCOCC1 Cc1cccnc1CCCNC(=O)C(=O)N(C)CCOC(C)CC(C)C c1(NC(=O)Nc2ccc(-n3nc(C)c(Cl)c3)cc2)nc(=N)[nH]c(O)n1 Cc1nc(NC(CCN(C(C)(C)C)C(C2OCCCO2)=O)=O)n[nH]1 c1(CC(N2CCC(NC(c3nc(Br)ccc3F)=O)C2)=O)c[nH]c2cc(Br)ccc12 c1(C(=O)NCC2CCN(C(C(C)(C)OC)=O)C2)ncn2ccc(C)cc12 C1(=O)C(CC(C)C)N1C1CC1.N1(CC(=O)OC)CCSCC1c1noc(CO)n1 C1(=O)CCCCCN1.N1(C(=O)Cc2ccc(C(F)(F)F)nc2)CCCCC(CO)C1 CC1(C)CCCC(C(=O)NC2CCC2NC(c2coc(C3CC3)n2)=O)CC1 C(C(C)(C)CN=[N+]=[N-])NC(CCC1(C)CCCN1C(=O)C(O)CC1CC1)=O c1(CN=C(NC(CC=C)CO)NCC2CCCO2)cnc2ccc(C)cc2c1 c1(-c2ccc(NC(C3(CC)CCOCC3)=O)nn2)ccnc(C#N)c1 c1(CC(=O)NC2CCC(NC(=O)C=CC3CCCO3)CC2)ccc2ocnc2c1 N1(S(CCOCC)(=O)=O)CC2CCC1CN2C(c1ccnc2[nH]nnc12)=O C1(NC(COC)=O)CCCN(C(=O)C(c2ccc(Br)cc2)C)CCC1 C1(C)(CNC(CC2C(C(=O)OC)C2(C)C)=O)CCN(C(=O)C(C)N(C)C(C)=O)C1 CSC=CC(=O)NC1(CCNC(=O)C(C)Cn2cccn2)CCCC1 N1(C(c2c(C)[nH]cc2)=O)CC(CNC(C2(c3cccc(Cl)c3)CC2)=O)C2(CC2)C1 Cc1cc(C(=O)NCC(C)CNC(c2ccoc2C2CC2)=O)cc(N)c1 Cn1cnc(=NC(=O)NCCC2CC(=O)N(c3ccc(Cl)c(F)c3)C2)[nH]1 Cc1cnccc1C(N1CC2C(NC(c3cccc(NS(C)(=O)=O)c3)=O)C2C1)=O C#CC1(C(=O)NC(C)CNC(=O)C(c2ccc(F)cc2)OC)CCCC1 C1(CNC(C2(CCC=C)CCCC2)=O)COCCN(C(=O)CCOC(C)C)C1 c1(-n2c(CN3C(CO)CC(c4ccccc4)CC3)cnc2)ccc(F)cc1F S(=O)(=O)(C1CCC(C)CC1)N1CCN(CC(=O)NC)C(=O)C1 c1(C2CCN(c3nnc(C(=O)OC)s3)C2)ccc(Br)cc1 c1(C(N2C(CNC(c3c(C)cccc3F)=O)C(C)CC2)=O)cc(O)cc(Cl)c1Cl N1(C(CNC(CC)=O)=O)CCCC2(C1)CN(C(c1c(C)nn(CC)c1Cl)=O)C2 Cc1oc(S(C)(=O)=O)cc1C(N1CCC(NC(=O)C(C)C(C)C)C1(C)C)=O c1(CCC(=O)N(C)CCN(C(=O)Cc2cnc[nH]2)C)cc(Cl)sc1Cl C#CCCCC(C)C(=O)N1CCC(C(N2CC(F)(F)CC2CC)=O)CC1 c1(OC)ccc(Cl)c(F)c1C(=O)NCC1CCCC1NC(=O)CC1(SCC)CC1 CCC(C)C(C(=O)NCCC1(C(=O)N(C(C)CN(C)C(C)=O)C)CC1)OC CCC(CC)C(=O)NC(CCNC(C1CCCN(C(=O)C(C)C)C1)=O)C(C)C CC1(C)CCCCC(C(=O)NCC2(C)CCCN2C(c2cc(N)ccc2Cl)=O)C1 N1(Cc2c(C)n[nH]c2)CC(F)(F)CC1CO.N12CCC(CC1)CC2=O c1(CN2CCC(F)(C(=O)Nc3ccc(CC)cn3)C2)c(C(F)(F)F)cccc1F c1(C(N2CCC(NC(CCN(CCC)C)=O)C2)=O)c(O)ccc(Cl)c1F N1(C(C(C(C)C)C)=O)C2CCC1CC(NC(=O)C(c1cccc(Cl)c1)(C)C)C2 N1(C(C2=NOC(C)C2)=O)CC2OCC(NC(c3csc(C(C)(C)C)c3)=O)C2C1 C=CC1CCCN1C(C1(C(=O)NCc2cn(CCO)nn2)CC1)=O CC12COCC1(C)CN(C(=O)CN(C1CC(C#N)C1)C(C1CC(C)(C)C1)=O)C2 c1(C(=O)NC(CCCNC(C(C)OCC)=O)C)ccc(Br)nc1N N1(C(C(C)C2CC2)=O)CCCC(CO)(NC(=O)COc2cccc(F)c2F)C1 c1(C(N(C(c2cn(Cc3ccc(O)cc3)nn2)C)C)=O)ccc2ncccc2n1 c1(OC)ccc(CN(C(=O)Cc2c(C)noc2N)Cc2cc(C)nn2C)cc1 CC1(C(=O)NCCC2CCC(NC(c3ccc(N)cn3)=O)C2)CCn2ccnc21 C1(NC(=O)CC2CCOC2)CC12CCN(C(c1cc(O)c(Br)cn1)=O)CC2 c1(NC(C2OCCN(C(c3c(OC)csc3)=O)C2)=O)ccc(Cl)c(O)c1 C1(COC)(NC(=O)C=CC2CCCO2)CCCN(C(C2COCCO2)=O)C1 N#Cc1ccc(C(N2CC=CC(NC(=O)CC3CCCN3C(N)=O)C2)=O)cc1 c1(C(=O)OC)c(C)[nH]c(C(N2CCC(NC(=O)C#CC(=O)NC)CC2C)=O)c1C c1(CCC(C)Nc2c(NCC)cccc2)nc2ccccc2[nH]1 N1(C(c2c(N)n(CCO)nc2)=O)CC2=C(C1)CN(C(=O)CCC1CCCO1)C2 C1(NC(C=CC=CC)=O)CCC(CNC(=O)CCc2cnc[nH]2)CC1 c1(N(C)C)ccc(C(N2CC(N(C)C)C(F)C2)C(=O)NC2CCC2)nc1 C1(CCC(N2C(Cc3cn(CCOC)nn3)CCC2)=O)CCc2ccccc2C1 N1(c2c(C(=O)OC)cccn2)CCC(NC(=O)CSS(C)(=O)=O)CC1C N1(C(C(C2(O)CN(C(c3c(C)cccc3F)=O)C2)F)=O)CC2CN(C)CC2C1 CCCC(C)(CCC)C(=O)N1CCC(NC(c2cc3n(n2)CCCN3)=O)C(C)C1 NC1CCN(C(c2cccc3sccc23)=O)C2(CC2)C1 N1(C(C(CC)OCC)=O)CCc2ccccc2C1CNC(C1CC2CCC1O2)=O N1(C(CCOCCC)=O)CCC2CCCC12C(N1CCCC1(CC)COC)=O C(=O)(C(O)CC(F)(F)F)NCC=CC(N1C2CN(C)C(C2)C1)=O C1(C(N2CCC(NC(CN3C(=O)C(C)C(C)C3=O)=O)C2)=O)CN2CCCN1CC2 C(C(CC(F)(F)F)NC(C1CCCCC(=O)N1)=O)NC(C1(CC(C)C)CC1)=O C#Cc1cccc(C(N2CCC(CNC(=O)CN3CCC(F)CC3)C(C)C2)=O)c1 C1(C(N2CCCC(NC(CCc3n(C)cnc3)=O)C2)=O)CC2(C)CC1CO2 C1(CNC(C(F)OC)=O)(NC(c2cccc[n+]2[O-])=O)CCCCCC1 C(N=c1nc(-c2cccs2)nc(N2CCOC3(CCC3)C2)[nH]1)C1(C)CCCCO1 c1(NC(C2N(C(CC(=O)OC)=O)CC3C2C3(C)C)=O)ccc(Br)nc1[N+](=O)[O-] Cc1cc(Br)cc(C(N2CCN(C(C3CCCN3C)=O)CC2C)=O)c1C c1(C(=O)NCC2C(NC(C3COCC3CF)=O)C2)csc(-c2ccco2)n1.C1CO1 C(CN=c1cc(NCc2ccc(C)cc2)nc(C)[nH]1)NCC(C)SC N1(C(C2C(C=C)CC2)=O)CCCN(CCNC(=O)CCc2nnc(C)n2C)CC1 c1(C(=O)NC2CCOCC2C(=O)NCC2CCCOC2)ccc2cccnn12 N1(C(C2CN(CC)C(=O)C2)=O)CCCC2(CCN(C(c3ccnnc3O)=O)C2)C1 N1(C(C2(COCC)CC2)=O)CCCC(CC(=O)N(C(C)CC(C)CC)C)C1 Cc1cc(C(=O)NC(C2CCCCN2C(c2ccnnc2O)=O)C)cc(N)c1 N1(C(C(CCC)C)=O)CC2CC(NC(c3cn4ncccc4n3)=O)CC1C2 C1(C(=O)OCC)(C(=O)NC2CC(O)(CNC(C3(CC)CCC3)=O)C2)CCCCO1 Cc1nocc1C(=O)NC1C=CC(CC(=O)Nc2sccc2C(N)=O)C1 N1(C(c2c(COC)cc[nH]2)=O)CCCCC12CC(NC(C1CCC(=O)N1C)=O)C2 C=CC1(CC(=O)NCC(CCOC)NC(=O)C(CC(C)C)N(C)C)CCCCC1 N1(C(CN(C(C)=O)C)=O)CC2CCN(C(=O)CN3CCCCC3)CC12 C(=O)(C1=CC(O)C(NC(=O)C(Cc2ccccc2)NCc2cccs2)C1)OC C1(C(=O)NC2CC(C)(CNC(c3cc(COC)cn3C)=O)C2)C2CC3C(C2=O)C13 c1(CCCC)ccc(C(=O)OCc2cccc(N3CCN(CC)CC3)c2)cc1N c1(OCCC(=O)NCC(N(C(C2C(=C)CC2)=O)C)C2CC2)c(C)cccc1C c1(OC)c(C(=O)NC2CCC3CC2CN3C(=O)CCC(F)F)[nH]c2ccccc12 Cc1nc(C(C)(C)C)[nH]c1CS(=O)(=O)N1CCC2CCC(O)C1C2 C#CC1CC2(CC2)CN1C(c1cc(CNC(c2c(C)cnn2C)=O)[nH]n1)=O CC1CCCn2c(C(=O)NCC3CCCN3C(=O)CCn3ccc(=N)[nH]3)cnc21 CCCC(C(O)C(=O)NCC(Cl)=CCl)NC(=O)C(CO)OC C(C)(C)(C(c1nnnn1C1CC1)NCc1cc(C2CC2)no1)OC CN1C2CCCC1CC(OC1CC(n3cc(C4CCCN4)nn3)C1)C2 C1(F)(CNC(=O)Cc2ccno2)COCCN(C(c2cc(Br)n[nH]2)=O)C1 N1(C(CC2C(C)CCN(C(CC(C)N(C)C)=O)C2)=O)CC2CCCC(C1)N2C c1(C(C)(C)C)ccc2cc(C(N3CCOC4CC34)=O)[nH]c2c1 C#CCC(C)C(=O)N(C(CNC(c1ccc(N2CCOCC2)nc1)=O)C1CC1)C c1(COc2ccc(NC(=O)Nc3c(C)cc(O)nc3)cc2)cnc2ccccn12 c1(-c2cc(C(=O)NC3C(NC(c4c(C)cco4)=O)CC3)no2)cccc(O)c1 CC(CN=c1[nH]c2ccc(Br)cc2s1)NC(C1CN(C)CC(C)O1)=O CCC(C)(CCC(C)C)C(=O)N1CC(C(C)NC(=O)CCS(C)(=O)=O)C1 CCC(C)CC(C)C(=O)NC1CC(NC(C2(N=[N+]=[N-])CC2)=O)C1 C1(CC(=O)N(CCCN(C(C(c2ccccc2)OC)=O)C)C)CCCCC1C C1(C(=O)Nc2scc(CCC(=O)OC(C)(C)C)n2)CCC(N)CC1 N1(C(C2CC(OCCN(C)C)C2)=O)CC(F)(F)CC1CNC(=O)Cc1cnc[nH]1 Cc1cc(CNC(C2CCN(C(C3CCC3(F)F)=O)CC2)=O)nnc1C N1(C(C=C(C)C)=O)CC2(CCC(CNC(=O)Cc3cn(C)nn3)O2)C1 N1(CC)CCCC(O)(NC(=O)CC2CN(c3cc(SC(F)F)ncn3)C2)C1 C1(C(N2CCOC(c3noc(C)n3)C2)C(=O)NCCOC)CCSC1(C)C c1(C(=O)NCCC2CC(NC(C(C=C)(C)O)=O)C2)cc(Br)c([N+](=O)[O-])s1 Nc1cc(C(=O)NC2CCN(C(=O)CCn3ccnc3)CC2CO)ccc1Br c1(N2C(C)CC(NC(=O)CN3CC4CCC3C4)C2)ncnc2ccc(F)cc12 N1(C(C2(CC)CCC2)=O)CCC(NC(=O)C(CCSC)NC(C)=O)C2(CCC2)C1 C(C(C(=O)NCC(CC)OC)C(C)C)NC(c1c(CC)cc[nH]1)=O Cc1nc(Br)c(C(=O)OC(C)CCOc2ccccc2)s1 C1(C)(C(=O)NCC2(CN(C(c3c(Cl)cn(CC)n3)=O)C)CC2)CCCCNC1=O N1(CC(=O)N(C(CNC(C2CCCO2)=O)C2CC2)C)C(=O)NC(C)(C)C1=O N1(C(CCC(CC)=O)=O)CCOC2CN(C(=O)CCC(C)OC)CC12 c1(C(COC)(C)O)cn(CCNC(=O)C(Cc2ccccc2)SC)nn1 c1(C(C(N2CCC(C(CC)CSC)(CC)CC2)=O)=O)cc(F)c(C)cc1Cl.OC c1(NC(C2(F)CN(C(c3cc(F)c(Br)c(F)c3)=O)C2)=O)ccc2c(c1)NCCC2 CC1COc2c(C(N3CC(F)(CNC(c4ncc[nH]4)=O)C3)=O)cccc21 C(=O)(C(F)(F)CCn1ccnn1)NC(=O)Cc1c(C(C)(C)C)[nH]c(=N)s1 c1(CC)nc(Cl)c(C)c(=NCC2CC(CNC(=O)CN3CCC(C)(O)C3)CO2)[nH]1 C=C(Cl)CC(C(=O)NCC1C(C)(C)C1(F)F)NC(c1cc(C)ns1)=O CC1(F)COCCN(C(=O)CC2C(NC(c3cn(CCO)nn3)=O)CC2O)C1 CCCCC(c1nnnn1Cc1ccccc1)NC(CC)C1CC1 C#Cc1cncc(C(N2CC(C(=O)NOCC=C(C)C)C(C)(C)C2)=O)c1 C(=O)(C1=CCCSC1)NC1CC(C(=O)Nc2cc(C(C)=O)ncc2)C1 N1(C(CC=C)=O)CCCC2(C1)CN(C(=O)C1=CC(C)(C)C1)C2 CC1CCCc2ncc(C(N3CC=C(CNC(C4CNC(=O)N4)=O)CC3)=O)n21 N1(C(C(c2cncnc2)C)=O)CCC2(CC1)CN(C(=O)C=CI)CCO2 CCC(CC(=O)N1CC(C)(OCC(=O)NCCC2CCOCC2)C1)C(F)F c1(C(C)=O)ccc(C(=O)NC2CC(NC(C3CC3C(F)F)=O)C2)cc1F C1(NC(COCC)=O)CN(C(c2cc(CC)ccc2O)=O)C2CCCCC12 N1(C(CCc2cc(C)n(C)n2)=O)CC(NC(=O)CC2COC(C)(C)C2)C(C)(C)C1 N1(C(C(C)Cc2ccnn2C)=O)CCCN(C(=O)C2=NOCC2)C(CO)C1 N1(C(c2ccsc2Br)C(=O)NCCC2CC2)CCCC1CCC(F)F.O c1(C(=O)NCC2N(C(CC3(COC)CC3)=O)CCCC2)cc2c(nc1N)CCC2 Cc1[nH]nc(C(=O)NCCC2CCCN(C(C3CCC(C(C)(C)C)O3)=O)C2)c1C CC(C)C(O)CC(=O)NC1(CO)CCCN(C(=O)Cc2cc(Cl)cs2)C1 C1(NC(c2ccc(OCC)nc2)=O)COC2(C1)CN(C(=O)CCNC(=O)CO)C2 C(CCC(=O)NCc1cc(C(=O)NOCCCCC2CC2)co1)=CC c1(C(=O)NC2CC(C)N(C(=O)C=C3CCCC3)CC2)cnn2ccnc(N)c12 C1(C)(NC(c2nc(CCC)oc2)=O)CCCN(C(=O)Cc2cc(C3CC3)no2)C1 CC1CCC(c2nnnn2-c2ccccc2)(NCCc2ccon2)C1 CC(N=c1[nH]c(=NC(C)CS(C)(=O)=O)c2sccc2[nH]1)c1nc[nH]n1 C1(C(=O)NCCN(C)CCO)COCCC1NC(=O)C=CC(F)F C=CCC(CNC(c1cc(O)n(CC)n1)=O)C(=O)N(CC(F)F)CC(C)O C1(C(N(C)CCNC(c2cc(Br)sn2)=O)=O)C2COc3ccccc3C12 c1(C(=O)NC(CC)CNC(c2c[nH]ccc2=N)=O)cc2c(cn1)CCCC2 C1(CNC(CCC=CCC=C)=O)CCN(C(c2cc(Br)cs2)=O)CC1C CN(CCCC(=O)NCC1CC(O)CN1C(=O)C=CC1CCCO1)N=O C12(C(=O)NCC3(CC)CCOCC3)COCC1CN(C(=O)CCN(C)C)C2 C1(C(=O)NCC(C)(CO)NC(C(CC)C)=O)CCN(C)CC1 N1(C(C)C(=O)N(C2CC2)CC2CC2Cl)Cc2ccccc2C1 CC(C)C(C(=O)NC1CN(C(C2CCC(F)C2)=O)C1)C(C)C c1(C(=O)NCCCCNC(CN(C(COC)=O)C)=O)cc(C)ccc1OC C(=O)(C1c2ccccc2C2CC1C2)NCC(C1CC1)NC(COCCSC)=O Cc1ccc(C(N2CC(NC(=O)CC3CCC(=O)N3)C(N=[N+]=[N-])C2)=O)c(N)c1C Cc1ccc(NCc2cc(C)[nH]c2C)c(CO)n1 C(=O)(CC1CCCc2oc(C)nc21)N1C2CC(CN(C(COCC)=O)C2)C1 Cn1c(C(C)(C)C)nc2cc(C(=O)NC3CCN(C(=O)C4CC4)C3)ccc12 n1(CCOC)cc(C(N2CCN(C(c3csc(O)n3)=O)CC2CF)=O)ccc1=O Cc1nnc2n1CC(C(=O)NCC1CC1NC(=O)C(C)(C)c1cccnc1)C2 c1(C(=O)NCC(CNC(c2ccc(N(C)C)cc2)=O)(C)O)cc(S(N)(=O)=O)co1 C1(NC(CSc2n(C)ccn2)=O)CN(C(c2cnncc2O)=O)CC1C1CC1 N1(C(C(C(C)C)C)=O)CCC2(CC1)C(NC(=O)C(C1CCCCC1)O)CS2(=O)=O c1(C(=O)NCC2CCN(C(Cc3c(C)non3)=O)C(C)C2)c(C)cc(Cl)cc1N c1(CC(N2CCC(NCC3CCC(F)(F)C3)C2)=O)cc(Br)cc(Br)c1 N1(C(CC2CCC(C)CC2)=O)CC2(CCC(NC(C3CC34CCC4)=O)CC2)C1 Cc1nc(CC2CC2)sc1C(=O)NC1CN(C(C23CC(F)(C2)C3)=O)CC1C N1(C(C(c2ccccc2)C)=O)CCC2CCC(NC(=O)CC3CN(C)C3)C1C2 c1(C(=O)NC2(C)CC(NC(=O)CC3CCCO3)C2)cc(Br)c2[nH]nnc2c1 Cc1onc(-c2ccccn2)c1C(N1C(C(=O)NC(C2CCC2)C)CC2CC12)=O C(C(C)C(=O)N1CCCC1C1CCN(C(=O)C(C)(C)OCC(F)(F)F)C1)OC N1(C(C(CC)F)=O)CCC2(CCC2NC(=O)CN2CCC(=O)NC2=O)CC1 CCCC(CC)C(=O)N1CC(F)CC1CN(C(=O)C(=O)N(C)C)C C(=O)(C1=CC2(CCOCC2)C1)NCC(CNC(c1c(C)nc(C2CC2)o1)=O)C c1(OC)cnc(Cl)c(C(=O)NC2CCCN(C(=O)C=C3CCOCC3)CC2)c1 c1(C(=O)NC(CNC(c2cc(C)nn2C(F)F)=O)C)ccc2c(c1)OCCO2 C(CCNC(C1CC1c1cccnc1Cl)=O)(C(C)C)NC(CNC(CC(C)C)=O)=O C(=O)(CCC1CCc2ccccc21)NCCN(C(C(C)=C1CCC1)=O)C c1(-c2cc(F)c(CN3CC4CC3CS4=O)cc2)ccc2c(c1)CCO2 CCC(CC)CC(F)C(=O)NC1CN(C(c2cnc(C)c(N)c2)=O)C2CCCC12 C1(C(N2CC(C)(NC(=O)COc3c(F)cccc3F)C2)=O)CCCNS1(=O)=O Cc1cccc(Br)c1C(C(C(=O)C(O)Cn1cncn1)=O)N.C1(CN)CCCS1 c1(CNC(C(C)NC(c2c(CC)n[nH]c2)=O)=O)cccc(CC)n1 CP(C)(=O)c1ccc(C(=O)NC2CN(C(=O)CCC3CCOC3)CC2F)cc1 C(=O)(C#CC1CCCO1)NCCN(C(=O)C(N1CCSCC1)C)CCC c1(N2CCC(F)(C(=O)Nc3cccc(CF)c3)C2)ncc2c(n1)CCC2 N1(CCCCCCCC)CCC2(CC1)CN(C(=O)C(C)NC(N)=O)CC(C)O2 C1(C(=O)NC2(CCCC)CCC2)(NC(=O)COCCCC(C)C)CC1(C)C Cc1cc(NC(C2CN(C(c3cc4cccnn4n3)=O)CCN2)=O)ncc1[N+](=O)[O-] C12CCCC(C1)NC2=O.C(C(=O)NCC1(CC(N)=O)CC1)N(CC)CC c1(OC)c(C)cc(C(N2CC(CNC(=O)C(Cl)=CCl)N3CCC2C3)=O)cc1C C(=O)(C(C)(C)C(C)(C)C)NCCNC(=O)COCc1nc(CC)on1 c1(C(=O)NC2CCC(NC(CCC(=O)N(C)C)=O)C2)cnc(O)n(C2CC2)c1=O c1(C(N2CC(CNC(C3C(C)C3C)=O)C2)=O)csc(-c2ccccn2)n1 c1(CC)ccc(C(=O)NCC2CC(NC(c3ccc(CO)o3)=O)C2)cc1F N1(CC=C)C(=O)NC(c2cc(C)cs2)C(C(=O)OCC)=C1C1CCOCC1 C12CN(C3(CCCCC3)C1)C(=O)C=CC(=O)N2.C=CCC(CC)C(=O)OCC N1(C(c2nc(OC)oc2)=O)CCCC2CN(C(C3(C(C)(C)C)CCC3)=O)CCC12 CCC(F)(F)CC(=O)NCCC1CCCCN1C(=O)CCc1c(Cl)cncc1Cl CC1CCC(NC(C2CN3CCC2CC3)=O)CN1C(C1(O)COC1)=O c1(-c2nc(NC(=O)NCC3CCCCC3F)oc2)c(F)cccc1F c1(C(C)NC(c2cnc[nH]2)=O)ccccc1OCC#N.C12CCC(C1)NC2=O c1(C(N(C(C)C)CCN(C)C(c2scnc2Cl)=O)=O)ccn2c1CSCC2 c1(C(N2CC(NC(C(c3cccc(OC)c3)C(C)C)=O)C2)=O)nccc(C)c1N C(CNC(C1CC(O)C1)=O)(CCNC(=O)C(C)N1CC(C)C1)OC CC(C#N)CN=c1[nH]c2c(c(=NCCc3nc(C4CC4)n[nH]3)[nH]1)CCCCCC2 c1(C(=O)NCC(C)CNC(=O)CC2C=CCC2)cc2c(nc1O)CCN(C)C2 c1(C(N(C)CC2CCCN(C(C(C(=O)OC)C)=O)C2)=O)nc(O)nc(O)c1F N1(C(CC(C)(C)OC)=O)CCN(C(c2n[nH]cc2Cl)=O)C(C)CC1C c1(C(NNC(CC2C(C)C2)=O)=O)cc2n(n1)CCCNC2=O c1(NC(CCOCCNC(CN2CC(CSC)C2)=O)=O)ccccc1C CC(C)C(C)CC(=O)NCCOCCCN(C)C(C1CCCC2(CC2)C1)=O c1(C(=O)NC2C(NC(C(CC=C)CC)=O)CCC2)[nH]c2ccccc2c1C1CC1 C(CCCC(=O)NCC(C1CC1)NC(c1cnc(-c2ccccc2)cn1)=O)SC CCCCCC(C(=O)NCCC(=O)OC)N1CCN(c2noc(C)n2)CC1 C(CCCCC(=O)NCC(C)(C)C1CCC1)N(C)C(c1cc([N+](=O)[O-])n[nH]1)=O CCC(C)(CC(=O)N(CCCN(C(=O)Cn1ncnn1)C)C)C(=O)OC C#CCCN=C(NCC(C)C=C)NCc1ccc(N2CCCCC2)c(C)c1 c1(C(N2CCC(CNC(c3n(CC)ncc3)=O)C2)=O)cc2cccnn2c1 c1(CC(=O)N(CC(CNC(CC2CC(OC)C2)=O)(C)C)C)ccc(Br)cn1 C1(NC(C=CC)=O)CCSC12CN(C(c1ccc(OC(C)C)cc1F)=O)C2 CCS(=O)(=O)CC(=O)NCC(C(C)C)NC(C1CC(C)(c2ccccc2)C1)=O C1(O)(CNC(C2CCN(C(C)=O)C2)=O)CCN(C(=O)Cc2c(C)n[nH]c2C)CC1 C1(C(=O)NC2CN(C(c3c(C)n(C4CC4)cc3)=O)CC2C)CCCNS1(=O)=O c1(C(=O)NCC2CC(CO)CO2)ccc([N+](=O)[O-])cc1.C12(CCCCC1)CN2 c1(C(=O)NCC(Cc2cccnc2)CO)cc(O)cc(O)c1 c1(OC)cc(OC)c(-c2ncc(C)c(C)n2)cc1CN1CCCC1C c1(C(=O)NC(C(C)NC(=O)CC2(CO)CC2)C)nccc2nn[nH]c12 N1(C(CC2(C)CCCCC2)=O)CCC(NC(=O)CCOCC(F)(F)F)C(O)C1 N1(C(CC2CCN(C)CC2)=O)C2CCC1C(C(=O)NCC1CC(O)C1(C)C)C2 N1(C(=O)OC(C)(C)C)CCCC1c1nc(CC2CC2c2cnsc2)no1 CC1(F)CN(C(=O)C=Cc2ccccc2)CCN(C(C2(O)CCOC2)=O)C1 CN=c1nc(N(CC(F)F)C)[nH]c(N2CCCC(N3CCCC3=O)C2)n1 C(=O)(C1=C(Cl)CCOC1)N1CCCC(NC(c2cnc(COC)s2)=O)CC1 N12CCCC(C3CN(C3)C(=O)c3c[nH]c(c3)C1=O)C2.C1(OCC)CC1C(C)(C)C C1(NC(C=COCC)=O)CCCN(C(=O)CNC(=O)C(C)CC)C1CC C(=O)(CCCC(=O)N(CCCOCCNC(C1(C2CC2)CC1)=O)C)OC(C)(C)C Cc1cc(C)c(C(N2CC3CC3(C(=O)NC3(CN4CCCC4)CC3)C2)=O)[nH]1 c1(SCNC(C2(O)CCN(C(=O)OC(C)(C)C)C2)C)cccc(C2=CCOCC2)c1 CC(C)C(O)C(=O)NCCC1COCCN1C(=O)C=CCN1CCOCC1 C1(C(=O)NC(c2c(OC)cccc2)CNC(=O)CCCF)CCc2ccccc2O1 c1(CC(=O)NC2C(NC(c3ncn(C(C)(C)C)n3)=O)C2)c(F)cccc1C#N C1(NC2CCN(C(=O)OC)CC2)CC2CCC(C1)N2S(=O)(=O)C1CC1 c1(C(=O)NCCC(C)NC(c2ccccc2C2CC2)=O)cnn2c1CCC2 CC1CN(C(=O)CNC(=O)Nc2ccoc2)CCN1C(=O)CSC1CC1 C(=O)(CCS(N)(=O)=O)NC.C12(CC=C)CCN(C1)C(=O)CC(C)CO2 Cc1cc(N)c(Br)cc1C(=O)NC(C)CN(C)C(c1cn(C)nn1)=O c1(C(=O)NC2CC(C)(C)N(C(=O)Cc3cccnc3O)C2)ccc([N+](=O)[O-])cc1 N1(C(c2nc(C)n(C(F)F)c2)=O)CCCN(C(C2CC2(Cl)Cl)=O)CC1C c1(NC(C2CC(NC(c3cncc(OC)n3)=O)C2)=O)cccc2[nH]nc(I)c12 N1(C(C(C(=O)OC)C)=O)CCC12CN(C(=O)C(C)Oc1ccccc1Cl)C2 c1(OC)cnc(Cl)cc1C(N1CCC(NC(C2(O)CCC2)=O)C(F)C1)=O C1(C(=O)NCC2(OC)CN(C(=O)C(c3ccccc3F)C)C2)CCCC(C)CC1 c1(C(=O)NC2(CO)CCN(C(C(CC)(C)C)=O)CC2)ccc(F)c2ncccc12 N1(C(Cc2c(C)nc(C)s2)=O)CC2(CCN(C(C34CCCN(CC3)C4)=O)C2)C1 c1(CNC(=O)NCC23CC(C(C)(C)C)(C2)C3)ccc2c(c1)C(=O)OC2(C)C C(=O)(CCCCCCCC)NC(CC#C)C(=O)NCc1cncn1C CCCC(C)CNC(=O)C(C)N(C(=O)CCCSCC)CCC c1(C(N2C(CN(C(=O)C(O)C(C)(C)C)C)CCC2)=O)noc2c1CCCC2 c1(C(C(=O)N(CC(C)NC(C2(CC3CCC3)CC2)=O)CC)C)ccnn1C n1(CC)ccc(C(=O)NCC2CCC2NC(C2CCOC2C(C)C)=O)n1 N1(C(CCC(C)(C)N(C)C)=O)CCC2CCCC12CNC(c1cccc[n+]1[O-])=O CC1(CNC(c2csnn2)=O)CCN(C(C2(C3CC3)CC2)=O)C1 N1(C(C(C(C)C)C2CCC2)=O)CC(CN(C(=O)CCC(F)(F)F)C)C2(CC2)C1 C1(CCCc2ccc(OC(CC)C)cc2)CCCN(C(=O)CC2CC2)CC1 Cc1nn(C)c(C(=O)NCC(CNC(=O)C(C)O)C(F)(F)F)c1Cl c1(C(N(C2CCN(C(=O)CC3CNC(=O)C3)C2)C)=O)c[nH]nc1F N1(C(C2N(C(c3c(OC)scc3)=O)C(C)C2)=O)CCC(N2CCN(C)C2=O)CC1 CC1CC(C)N(C(=O)CNC(=O)C(F)(F)F)CCN1C(=O)CCc1cc[nH]n1 c1(C(N2C(CCCNC(CSCC)=O)CCC2)=O)cc(Br)cc(C)c1F c1(C(=O)NCCCN(C(C2C(CC)C2)=O)CC2CCCC2)ccc(F)cc1F Cc1cc(C(=O)NC(C)CC(C)NC(=O)Cc2ccc(F)cn2)nc(N(C)C)n1 CC1CCCC(C)N(C(C23CC(NC(C4CCCCS4)=O)(C2)C3)=O)C1 c1(CC(N2CC(N(C)C(c3n[nH]cc3N(C)C)=O)C(F)C2)=O)ccc([N+](=O)[O-])cc1 C1(C(N2CC(CCOC)(OC)C2)=O)CN(C(c2cccc[n+]2[O-])=O)C(C)(C)C1 c1(-c2cn(CC(N3CCN(CC(=O)NCC#C)CC3)=O)nn2)ccc(Cl)cc1F c1(C(=O)NC2CN(C(Cc3ccc(SC)cc3)=O)C2)cc2c(s1)CCS(=O)(=O)C2 N#Cc1ccc2c(=NC(=O)C3CCCC3NCc3cc(O)cc(F)c3)[nH][nH]c2c1 C1(c2cn(CC(CN(C)C)(C)C)nn2)(NC(c2c(OC)n[nH]c2)=O)CCCCC1 n1(CC)cc(C(=O)N(C2CCN(C(=O)CC3CC(=O)C3)C2)C)nn1 C12(O)CCCN(C1)C(=O)C(=O)NC2.C(F)(F)(C(F)(F)F)OCC(=O)N.CNC C1CCN1C(=O)CC1CC1.C(C(=O)N(CCCCC)C1CC1)N(C(=O)OCC)C.C1CC1 c1(C(=O)NC2C(CNC(c3ccc(O)nc3)=O)C2)cnccc1Br N1(C(COCC(=O)OC)=O)CC2CC1CCC2NC(c1sc(CO)nc1C)=O CC1=CCC(C)(C(N2CCN(C(=O)C=Cc3ccc(Cl)cc3)C(CF)C2)=O)CC1 CC1COc2c(C(=O)OCC3CCc4cc(Br)ccc4O3)cnn2C1 N1(C(C(C)C#N)=O)CCOC(Cn2cc(C3CCCCC3)nn2)C1 C(=O)(C1=CC2CCCCCC12)NCC(C1N(C(CCC(C)(C)O)=O)CCC1)(C)C N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CC1)CC2C(=O)NCC1COC(=O)N1 N1(C(CCC)=O)CCC2C(C1)CN2C(c1cc(C2CC2)nnc1O)=O C1(C(F)(F)F)(NCCF)CC2CCC1C2.c12ccccc1C(C1CC1)NC(=O)C2 O=C1CCCN(C(C23CSCC2C3)=O)C(c2ccccc2)C1 Cn1nccc1C(F)=CC(=O)NCC1COCCN(C(=O)Cc2cncs2)C1 Cc1ccc(C(=O)NC(C)CCNC(C2(C#N)CC(C)C2)=O)c(C)c1 C(C1CCCCC1)=CC(=O)NC1(CC(C(=O)NCCOCCCN(C)C)C)CC1 N1(C(c2cncc(N(C)C)n2)=O)CC(C2CN(C(=O)Cc3ccc(Cl)s3)C2)C1 C(=O)(C1=CSCCO1)NC(c1ccccc1)C(C)NC(=O)C(C)(F)F c1(C(=O)NCc2cc(C(N(C(CCCC)C)C)=O)on2)cc(CC)oc1C C1(C(N(C(C)CN(C)C(=O)OC(C)(C)C)C)=O)CCC1S(N)(=O)=O c1(C(=O)NCCNC(c2cccc(C)c2C(F)(F)F)=O)cnc2c[nH]nc2c1 c1(C(N2C(C)C(C)N(C(=O)CNS(C)(=O)=O)CC2)=O)cccc2c1CCCC2 C(=O)(C(F)C(=O)NCC1(C)CCCN1C(=O)C(c1ccccc1)F)OCC c1(-n2cc(C(N3CCC(CSCC)C3)=O)nn2)ccc(NC)cn1 Cc1cc(CC(=O)NC2CC(n3cc(C(C4CCCC4)C)nn3)C2)n(C)n1 N1(C(=O)CC2CC=CCC2)CC2CCC1CN2C(=O)CC1CC2(CCC2)CO1 C1(NC(CCC#N)=O)CN(C(=O)CCOc2cc(Cl)cc(Cl)c2)CC12CC2 c1(C(N2CCCC(C(=O)Nc3cc(F)ccc3F)C2)=O)ccnc([N+](=O)[O-])c1 C(C1=NOC2CN(C(=O)CCC(F)(F)F)CC12)NC(c1ccc(COC)o1)=O C(N=c1nc(NCC2CN(C3CCC3)C2)c2c([nH]1)CCS2)C1CCCO1 N1(C(c2scc(C(C)=O)c2)=O)CCC(C)(C)C1CNC(C1CCC(C)CC1)=O Cn1c(O)ncc(C(N2CCC(C)(NC(C3CCS(=O)(=O)C3(C)C)=O)C2)=O)c1=O c1(SC)nc(O)c(C(=O)NC(C)CN(C(=O)CC2CCC(C)(C)C2)C)cc1C#N C1(NC(Cn2c(C)cc(C)n2)=O)C2CCC1CN(Cc1ccc(Cl)c(I)c1)C2 C(=O)(CC(C)(C)C#N)N(CCC(=O)NCC1CC1C)CC=C C(=O)(CCCCC(=O)c1ccc(OCC)cc1)NC(c1nc(=O)o[nH]1)CC C1(C(=O)NC(CN(C(c2c(CC)cc[nH]2)=O)CC)C)CCCS(=O)(=O)C1 c1(NC(=O)OC(C)(C)C)cc(CO)ccc1Br.c1(N)ccnn1Cc1nc[nH]n1 c1(CC(NOCC(=O)NC(C)Cc2ccccn2)=O)ccc(O)nc1 C1(CC(C)C)(NC(C2(CNC(=O)CC3CC(F)C3)CCC2)=O)CCCC1 N1(CCCC)CCCCC1C(=O)NCC1CC1NC(=O)C(O)C1CC1 CCC(C(=O)N(CC(C)NC(c1nonc1N)=O)C)n1ccnc1 N1(C(C(C)OC)=O)CC2CC2(C(=O)NCc2ccc(OC)nc2)C1 c1(CNCC(C)OC(C)(C)C)ccc(S(=O)(=O)NC2COCC2O)cc1Br c1(N2C(CNC(Cc3c(C)nn(C(C)C)c3C)=O)CCC2)ncccc1S(C)(=O)=O c1(CNC(C2C3CC2N(C(C2(C4CC4)CC2)=O)C3)=O)ccc(Cl)c(Cl)c1 N1(C(CC2N(CC)CCC2)=O)CCC(NC(=O)CC2(O)CCC2)C12CC2 C1(C2CC2)(NC(CN(C)C(N)=O)=O)CCN(C(=O)Cc2cnc[nH]2)C1 N1(C(C2(CC=C)CC2)=O)CCC(CNC(C2(CCF)CCOCC2)=O)C(C)C1 c1(C(=O)NCCN(C)C(c2ccncc2F)=O)cc(-c2ccccc2)nc(O)c1 CC(C)C(CNC(=O)CC1OCCO1)C(=O)Nc1cncc(C2CC2)c1 O(NC(=O)CC(CC)NC(C1CC(O)C(F)C1)=O)CC(=O)OCC N1(C(C(CC)OCC)=O)C2CCC(C2)C1C(=O)NCC(F)(F)C(C)C O(N(C)C(=O)CNC(=O)COCCNC(C1(C#N)CC1(C)C)=O)CC C(CCCCC(=O)NOCc1nc[nH]n1)N(C(CC1(OC)CCC1)=O)C N1(C(C2CCC(C)(CC)O2)=O)CCC(C2CC2)C1CNC(c1sc(O)nc1O)=O C=C1CCN(C(=O)C=C(CC)CC)C(C(=O)NCCN(CCCF)C)C1 N1(C(C(C2CCOC2)OCC)=O)CCC(CNC(c2cc(C)n(C)n2)=O)C12CC2 C1(NC(C(C=C=C)C)=O)CN(C(=O)CNC(C2CCC2)=O)C2CCCCC12 C1(NC(=O)C=CCN2CCCC2)COCCN(C(C23CCC(CC2O)C3)=O)C1 Cn1c(C(=O)NC2CCC(NC(=O)CCCC3CCCC(=O)N3)C2)cnc1Cl Cc1cccn(CC(=O)NC2COCC2NC(=O)CC2CCCSC2)c1=O C1(CC(=O)NC(C2CC2F)=O)CCCC12CN(N1CCC(O)C(F)CC1)C2 c1(C(=O)NCC(CC)NC(=O)CCCC(C)(F)F)cc2ccncc2[nH]1 Cc1cccc(C)c1CC(N1CCC(F)(CNC(c2nc(C)n(C)n2)=O)C1)=O C(=O)(CC(O)C(Cl)(Cl)Cl)NCC(CN(C(c1ccc(SCC)cc1)=O)C)C C1(CC(=O)N(C2CCN(C)CC2)C)CC(C)(C)CN1C(C1CNC(=O)O1)=O N1(C(CC=CC=C)=O)CCN(C(=O)C(O)C2CC2)CC1CO C1(NC(C2CC(=C)C2)=O)COCCN(C(c2[nH]cnc2C)=O)C1 C1(NC(CSSC)=O)(COC)CCN(C(=O)CC2CCCN2C)CC1 CC1(CNC(=O)C(Cc2cn[nH]c2)NC(=O)CCc2ccoc2)CCOC1 C1=NCC(CCNC2CCCCC2)(S)C1.c1(C)nc(C2COC2)no1 c1(OC)cc(F)c(F)cc1C(N1CC(CNC(C23CCC(C2)C3)=O)C1)=O c1(OC)cccc(OCC(=O)NC2CCN(C(c3cc(Cl)cn3C)=O)CC2)c1 N1(c2ccc(NC(=O)NCC)cc2)CCC(C)(OC)CC1.N12CCC1C2 CC(=Cn1ccnn1)C(=O)NCC1CN(C)CCN1c1cc2nncn2cn1 c1(C(=O)NCC2CN(C(c3c(CC)ncnc3)=O)C2)cn2cc(Cl)cc(Cl)c2n1 c1(CN2C(C(N3CCn4nccc4C3)=O)CC(O)C2)cnc2c(Br)cc(Cl)cn12 N1(C(c2cnc(CCCCC)o2)C(=O)NCCSC)CCOC2COCC2C1 c1(NC2C(NC(C(CCC)OC)=O)CCCC2)cc(C(C)(C)C)nc(C(C)C)n1 Cc1cc(-c2cn(C(C)CNC(C3(C)CC3(F)F)=O)nn2)ccc1Br CCC(C)(C(=O)OC)C(=O)NCCCNC(=O)CNC(C)=O c1(CCC)c(C(=O)NCC2CCCCC2NC(=O)C(C)SC(F)(F)F)nnn1C Cc1cccc(Cl)c1NC(=O)COC1(C)CCC1.N12CCC(C)(C1)CCC2=O CC1CCCC1(c1nnnn1-c1ccc(F)cc1)NCCCSC(F)F c1(CCCC(=O)NCC2CCCN(C(=O)C(F)n3ccnc3)C2)ccc(Cl)cc1 c1(C(N(CCN(C(C2C(CC)CCCC2)=O)C)C)=O)c(C)ccc(C)c1N N1(C(CCCCNC(C(CC=CC)CC)=O)=O)CC2OC(=O)N(C)C2C1 C(=O)(CC(c1ccccc1)N(C)C)NC1C(NC(C2C(C(C)(C)C)C2)=O)CC1 c1(CNC(C(c2ccc(N)cn2)(F)F)=O)cccc2c1CNCC2 N1(C(CCCCCC=C)=O)C(CNC(=O)CCc2ncco2)CC2CCCCC12 C1(C2(O)CN(C(=O)CCS(C)=O)C2)(CNC(c2n(CC)c(O)nc2)=O)CC1 CC1=CC(NC(C2(C)CCCN2C(=O)CC2NC(=O)NC2=O)=O)CCC1 C1(CCNC(C2(C)CN(C(CCC)=O)C2)=O)CCOC(C)C1 CCC(C)CCC(=O)NCC1CN(C(=O)CC2CCSCC2)CC1(C)C CC(CN(C)C)CC(=O)N1CCC(C(=O)N(CC(C)(O)C2CC2)C)CC1 C(=O)(CCC(C)(C)C)NCC1CCN(C(C2(CC)CCCO2)=O)C1 C#CCCCCCNC(C1(NC(c2c[nH]c(=NC)o2)=O)CCC1)=O C(=O)(CC(C(F)F)NC(=O)C1=CCSC1)NCC1(C(C(C)C)O)CC1 C(CCCCC(=O)N(C1CCCN(C(C2CCCCC2(F)F)=O)CC1)C)N(C)C c1(C(C(=O)NC2C(NC(C3C(CC)CCO3)=O)CC2)(F)F)ccc(C)cc1 c1(C(N)=O)cccc(N2CCN(C(c3ccc(CCCCCl)o3)=O)CC2)n1 c1(C(N(C(C)CCNC(C2CC2C#N)=O)C)=O)cc(C(F)(F)F)cc(Br)c1 CCC(CC)CCC(=O)NC(C(=O)NC1CCC(C2CC2)C1)C(C)(C)C Cc1cc(P(C)(C)=O)oc1C(N1c2ccccc2CC1C)=O C1(F)(COC(C(C2CCCCCC2)C)=O)CCCCC1 C1(C(=O)NCCCC(C)NC(C=CC(C)(C)SC)=O)CCc2c(ncn2C)C1 CC1CC(NC(=O)C(=O)NC2CC2)CN(C(=O)CCCCc2ccc(F)cc2)C1 c1(-c2onc(-c3nc(C)sc3)n2)cc2c(s1)CCC(C)(C)C2 N1(CC(=O)OC)CCCCC(NCc2cccc(C)c2-n2cccc2)C1 Cc1ccc(Br)c(F)c1C(=O)NCC1(O)CCCN(Cc2ccc(O)cc2Br)C1 C1(NC(C2CCC(C)(CC)O2)=O)CN(C(c2cccc(N)n2)=O)C2CCCCC12 c1(C(N2CCN(C(C3CC4(CC(=C)C4)C3)=O)C3C2C3)=O)ccn2c(O)nnc2c1 C1(NC(c2c(C)nc(C(C)C)s2)=O)CC2CN(C(c3cnccn3)=O)CC12 CCS(=O)(=O)CCCCCN1CCC(NC2CNC(=O)CC23CCC3)CC1 C(=O)(C(C(C)(C)C)N1CCCC1=O)NC(CN(C(c1c(CC)cno1)=O)C)C c1(CC)ccc(OC)cc1OC.C12CCCCC1C(=O)O2 CCCCC(C(=O)N1CCCC(F)C1)NC(c1ccc(Cl)s1)=O c1(C(=O)NCC(CNC(=O)C(O)Cn2cncn2)OC)cc2c(cn1)OCCC2 c1(C(N(C2CCN(C(CCC(C)C)=O)C2)C)=O)cnn2c1C(=O)NCC2 Cc1cc(C(=O)NC2CC(CC(=O)NCC(CO)C(C)(C)C)C2(C)C)nnc1O c1(OC)cc(C(=O)NCCN(C)C(C2CC2CF)=O)c(F)cc1N c1(CN(C)C)ccsc1C(=O)NCCOC1CN(C(=O)CC2CC=CCC2)C1 C(c1cnccc1C)=CC(=O)N(CC(CC)NC(=O)C#CC1CC1)C CC(C)(CNC(C1CCCC(NC(=O)CCC2CCC2)CC1)=O)CC(F)F C(=O)(CCCCCF)N1CCCC(N(C(c2cc(-c3ccc(C)o3)[nH]n2)=O)C)C1 c1(C(N2CCC(C(C)NC(=O)CCc3cnco3)C2)=O)cc(Cl)ccc1F C1(NC(c2ncn(C(C)C)n2)=O)CN(C(c2nccnc2Cl)=O)CC1O c1(C(N2CCC(C(=O)NC3CCCCC3CCO)(CC)C2)=O)ncnc(O)c1F C(C(C(=O)NCCC(C)N(C)C)C(C)C)NC(c1cncc(OC)n1)=O N1(C(COC(CC)C)=O)CCC(CO)(CNC(c2sc(C)cc2C)=O)C1 O=C(N=c1nc2c(F)cccn2[nH]1)N1CCOC(c2ccccc2Cl)C1 C1(NC(c2c(C)n(CCO)cc2)=O)C2CC3CN(C(=O)CCF)C1C3C2 N1(CC(=O)NC23CC(CNC(C(C)(Cl)Cl)=O)(C2)C3)CSCCSC1 CCC(C)CCC(=O)NCCNC(=O)Cn1cc(C(F)(F)F)ccc1=O N1(C(C(C(C)C)CNC(=O)Cc2cnnn2C)=O)CC2(COC(=O)N2C)C1 N1(C(C2(O)CCN(CCN(C)C)CC2)=O)CCc2cnccc2C1 Cc1c(F)ccc(C(=O)NCC2CC2CNC(C2(C3CCCO3)CCCC2)=O)c1Cl C1(COC)CN(C(=O)CCC(C)(C)N(C)C)CCN1C(=O)C1CC1 c1(NCc2c(Cl)cn(C)n2)ccc(S(=O)(=O)NCCc2cn(C)nn2)cc1Br Cn1c(C(N2CCC3(CNC(=O)C=CCO)CCCC23)=O)cc2sccc12 N1(C(C(C)OCC(C)C)=O)CCCN(C(c2cccc[n+]2[O-])=O)CC1CO Cn1cc(CC(=O)NC23CCN(C(=O)CCC(C)(F)F)CC2C3)c2ccccc12 C1(CCNC(=O)CC23CC(C2)C3)CCCN(C(c2n[nH]cc2Cl)=O)C1 C1(CNC(C2CCC(C)(C)C2)=O)CCCC2CN(C(=O)Cc3csc(Cl)n3)CC12 C(=O)(CCC(C)(C)C)NCCC(C)(C)N(C)C.c12ncc(cn1)[nH]2.C1CO1 c1(OC)noc(C)c1C(=O)NCC(N1CCN(C(=O)C=CSC)CC1)C(F)F Cc1ccc(CC(=O)NC2CC(C)N(C(=O)CCc3ncc[nH]3)C2)cc1F C1(NC(C=CCCC)=O)CCC(C)(CNC(=O)CN(C2CCS(=O)(=O)C2)C)C1 CCC(CNC(c1cc(C(N)=O)c[nH]1)=O)N=c1[nH]c(Cl)ncc1[N+](=O)[O-] N1(CCC(N2CCC3CN(C(COC)=O)CC2C3)=O)C(=O)Cc2ccccc2C1=O c1(C(=O)NCC(=O)Nc2cccc(CC)c2)ccc2c(c1)CCN2S(C)(=O)=O n1(CC)c(O)nc2ccccc12.n1(CCC#C)c2nnc1C(F)(F)C1CCN2C1 c1(C(N(CCC(C)NC(C2(C)CCC2)=O)C)=O)cnc(Br)s1 C=CCC(CC(=O)NCC1CCC(CO)O1)NC(C1CCC(C2CC2)C1)=O c1(C(C)OC(=O)C(C)COC(N)=O)cccc2ncccc12 N1(C(C(CCC)OC)=O)CCN(C(c2nc(O)sc2C)=O)CCC1C CC(C(=O)NC1CC(CCNC(c2cnn(C3CCOC3)n2)=O)C1)C(F)F N1(C(C(N)=O)=O)CCN(C(C2CCN(C(=O)NCCCl)C2)=O)CC(O)C1 C12(C(N(C)CC3COCCO3)=O)CC(CO)(CN1C(=O)C#CC1CC1)C2 C1(NC(CNC(CN(C)C)=O)=O)CC(F)(CNC(=O)C(F)(F)c2cncs2)C1 N=c1cc(C2CCN(C(C3CCCN3C3CC3)=O)C2)c(O)n[nH]1 Cc1ccc(OCCC(=O)NCC2CCCC2NC(=O)CCSC(=N)N)c(C)c1 CC1(C)CC(NC(C2CCC3(CC3)N2C(=O)CN2CC=CC2)=O)C(=O)O1 CC1C2CC(C2NC(=O)C(C)(C)N2CCOCC2)N1C(=O)CN(C)S(N)(=O)=O CN1CC(C(=O)NC2CCC(CC(=O)N(CCCO)C)CC2)CCC1=O S(=O)(=O)(c1cccc(Br)n1)C(C1CC1)=O.c1(N)ccn2cnnc2c1 N1(C(CC=CC(C)(C)C)=O)CCN(C(=O)COc2cccc(Cl)c2)CC(O)C1 C(CCCC(CO)NC(=O)CCCCC1CC1)NC(COc1cccc(C)c1)=O C1(NC(C(CN(CC)CC)F)=O)(CC)CCCN(C(C2C3CC(=O)CC23)=O)C1 C1(NC(C(c2ccccc2F)C)=O)CN(C(=O)CCN(S(C)(=O)=O)C)CC1O Cc1csc(NC(c2cc(-c3ccccc3)ccn2)=O)c1Br Cc1nc(NCC2C3CN(C(c4ccc(Cl)cc4Cl)=O)CC23)ncc1[N+](=O)[O-] C1(C(=O)NC2CC(CC)(CC)C2)CN(C(C2CCO2)=O)CCN1C CC1(C)CCCC(NC(=O)Nc2nc(C(F)F)cs2)CC1 N#Cc1cc(C(=O)NC2CN(C(c3cc(O)cc(Cl)c3)=O)CC2C#N)ccc1F c1(C(=O)NCC#CCNC(C(C)O)=O)ccc2nc(Cn3cncn3)[nH]c2c1 C1(C(=O)NC2C(NC(c3c(C)con3)=O)CCCC2)CN(CP(C)(C)=O)C1 S(=O)(=O)(c1cnc(NCC(C)C(F)F)c(Cl)c1)NCC1(CC)CCOC1 N1(C(CC(C)F)=O)CCC(F)(CNC(=O)CCCc2cccc(Cl)c2)CC1 c1(C(N2CCC(NC(C3OCC(C)C3)=O)C2C)=O)cc(O)nc2c1CCCN2 CC(C)C(O)C(=O)NCC1CN(C(c2cn(Cc3cccs3)cn2)=O)C1 N1(C(=O)CCc2ccsc2Cl)CCCCC2(CCN(C(=O)CC3CCCO3)C2)C1 n1(CC(=O)NC2C(NC(C3C(C)(C)S(=O)(=O)CC3)=O)C2)ncn2cccc2c1=O CC1CCC(=CC(=O)Nc2nc(Cc3cccs3)cs2)C1 C1(C(N2CCCOCC2)=O)CC(F)(F)CN1C(C1CCCS1)=O CS(=O)(=O)C1(C(=O)NCC2CCC3CNCC3C2)CCCCC1 O=C(CCCc1cnccn1)N(C1CSC1)CCO C1(CC)CN(C(=O)C(F)(F)c2cnnn2C)CCC1NC(=O)CCCNC(C)=O C1(NCC2(CN(C(c3c[nH]nc3C(F)(F)F)=O)CC3CC3)CCC2)CS(=O)(=O)C1 c1(C(N(CCC(=O)N(CCCN=[N+]=[N-])CC)CC=C)=O)c(CO)n[nH]c1C Cc1nc(=N)[nH]cc1C(=O)N(C)CC1CCCN(C(=O)CCCCC2CC2)C1 N#Cc1cc(=NCC2CCC3CC2CO3)cc[nH]1 C1CC(C(C)C)O1.C(C(C(=O)N1CCC1CC(N)=O)n1cc(CC)nn1)OCC C(CC1=CCN(C(=O)CCN(CC(F)(F)F)C)CC1)NC(C1ON=C(CC)C1)=O C1(CNC(C(CC2CC2)OC)=O)CCN(C(c2ccc(O)cc2F)=O)CC1(F)F Cc1ccc(Cl)c(C(N2CC(NC(c3cnc(C(F)F)s3)=O)C3CC23)=O)c1 N1(C(C(OC)OC)=O)CCC(c2ccccc2C(N2CCC(CO)C2)=O)CC1 N1(C(CN2CC(C)(OC)C2)=O)CCC(NC(c2cnncc2C)=O)C1C(C)(C)C Cc1cnc(C(=O)NC2(CCC(=O)N(CC(C)(O)C3CC3)C)CCC2)cn1 c1(C(=O)NCC(C)(O)CNC(c2cc(O)cc(=O)o2)=O)ccnc2ncnn12 CC(C)CCC(F)C(=O)N1CCOC(CC(=O)Nc2ccc(Cl)cc2)C1 C(C)(C)(CCCNC(=O)CC1CC=CC1)NC(C(C)N(C(C)=O)C)=O C(c1ccsc1C(F)(F)F)=CC(=O)NC1CCC1NC(=O)Nc1cccc(F)c1 c1(CN2CC(Nc3nc(OC(C)C)c(Br)cn3)C(C#N)C2)c(F)ccc(C)c1F C1(NC(C(=O)NCC2(N(C)C)CC2)=O)C2CC3CC(C2)CC1C3 Cc1ccc(C(N2CC3CC2C3C(N2CCCC(C)C2CO)=O)=O)c(I)c1 c1(C(N2CCC(N(C(=O)C=Cc3cnn(C)c3)C)C2)=O)ccc(C(F)F)cc1Cl N1(C(CC(C)OC)=O)CCN(C(=O)CC2C(=O)ON=C2C)C(C2CC2)C1 c1(CNC(c2n(CC)nnn2)c2cccnn2)ccc(Cl)cc1 C1(NC(=O)CNc2ccccn2)CCCCCC1NC(c1coc(C2CC2)c1)=O C#CCCCC(=O)NCC(CC)N(C(=O)C(C(C)C)Sc1ccccc1)C N1(c2ccnc(NCC3C4(CC(C)(C)C4)C3)n2)CC2CC3COCC3C2C1 C12(C(N3CC(CN(C(C)C(N4C(=O)CCC4SC)=O)C)C3)=O)CCCC1OCC2 c1(N(C)Cc2c(F)cccc2Br)ncnc2c1ncn2C1COCCC1(F)F C1(NC(CC(C)SC)=O)CN(C(C2(CO)CCOCC2)=O)CC12CCC2 C1(C(=O)NC(C)CCCCNc2nccnc2C#N)CCC2C(C1)C2(F)F CCCC(C#N)C(=O)NCC(C)C(N1CCC(C#N)CC1)=O Cc1cc(CC(N2CCCCC2CCNC(C2CC(C)(O)C2)=O)=O)ccc1Cl N1(C(c2c(Cl)cn(CC)n2)=O)CCC2C(C1)CN2C(=O)C(C)c1ccco1 Cc1cccc(CN(C(=O)CC(O)CNC(=O)C(C)C2CC2)C)n1 N1(C(C(CC)C)=O)CC2CCCN(C(c3ccccc3)C3CCCCC3)C2C1 C(CN(CC(O)CN(C)C)C)(C(C)C(C)C)NC(C)Cc1ccccc1 c1(C(N2CCN(C(CCC#C)=O)CC2CC2CC2)=O)cnc2nc(O)ccc2c1 CC(C)(C)CC(F)C(=O)NC1CC=CCC1C(=O)NCCn1cc(CO)nn1 c1(N2CCCC(OCC)C2)ncc(C)cc1S(=O)(=O)NCC(CO)C1CC1 CCC(C)C(O)C(=O)NCCCCNC(c1cnoc1C)=O C(CCCCCN)(OC)OC.C(CC(F)(F)COCC)C1CCN(CCOCC)C1 C(=O)(C(C)(C)C(C)(F)F)NCC1(NC(c2cc(OC)c(O)cc2)=O)CCC1 C=CCCCC(C(=O)NC1CC2(CCC2)C1O)NC(C1CC(=O)CC(=O)N1)=O c1(CNC2(c3nnnn3C)CCCC(C(C)C)C2)noc2cc(F)c(F)cc12 N1(C(c2ccc(CSC)o2)=O)CCCC1(C)CCC(N1CCC(C)(O)C1)=O N1(C(=O)Nc2cc(CC(=O)OC)[nH]n2)CCc2ccc(OC)cc21 N1(C(c2cc(CCC)on2)=O)CCOCC(F)(CNC(c2ccc(OC)o2)=O)C1 N1(C(C2C(CCC)C2)=O)CCC2(CC1)CN(C(c1nsc(OCC)n1)=O)C2 C1(C(=O)NCCC(CC)(F)F)CCN(C(=O)CCC(C)C)CC1(C)C CC(CC(=O)NCC1C(CNC(=O)C(C)S(=O)(=O)C(C)C)C1(F)F)CC(F)(F)F C1(OC)CC2CCC1CC2C(=O)NCC(CO)NC(c1nccc2occc12)=O c1(C(N2CCOCC(CNC(=O)CSCC(F)(F)F)C2)=O)cc(F)cc(F)c1F N1(C(C(CC2CN(C(=O)CC3CC(CF)C3)C2)F)=O)CCC(F)(F)C(F)C1 C1(C(N2CC(NC(C=CC(CC)C)=O)C(OC)C2)=O)CC2(C1)CC21CC1 N1(C(CC2CCCC(C)(C)C2)=O)CCC(CNC(c2cnco2)=O)C(F)(F)C1 Cc1sc(NC(=O)COC(C2CCOC2=O)=O)nc1-c1cccc(F)c1 C=CC(C)(O)CC(=O)NC1CC2(C1)CC2NC(C1C2(CC2)C12CC2)=O C1(CN(C)C(c2ccn(C(C)(C)C)c2)=O)CCCN1C(=O)CCc1cnc(O)[nH]1 Cn1cc(NC(C2(CNC(=O)CC34CCCC3C4)CC3(CC3)C2)=O)c(Cl)n1 C(=O)(C1=CCCSC1)N1CC(SC)C(NC(=O)CNC(c2ccncc2)=O)C1 c1(C(C)=O)ccnc(C(=O)NCC2C(C)CCN2C(=O)CCOC2CCCC2)c1 N1(C(C(CCCCC)CC)=O)CCCCC(C2CN(C(c3sccc3F)=O)C2)C1 c1(C(N2CCN(C(C(COC)C)=O)CC2C)=O)ccc(S(N)(=O)=O)s1 c1(N(CCOC(COC)C2(C)CC2)C)nc(OC)ccc1Cl.C(C(=O)N)(C1CC1)OC Cc1cc(=O)c(C(N2CCOC(CC(N3CCCC(OC(C)C)C3)=O)C2)=O)c[nH]1 C1(C(=O)OC(C)CCc2cn[nH]c2)CCN(C(=O)OC(C)(C)C)CCO1 c1(C(=O)NCC(C)NC(C2C(C(=O)OC)C2)=O)cn(CCc2cccs2)nn1 C=CC1(CNC(=O)C(C)CNC(=O)CCC2CCOC2)CCOCC1 C1(NC(CCCC2C(C)C2)=O)CCCC(NC(c2cn(C)nc2Br)=O)CC1 c1(C(=O)NC2CC3(CC(NC(C4(C)CCOC4)=O)C3)C2)ccc2c(c1)CCOC2 C1(CNC(C2(C=C)CCC2)=O)CN(C(c2cc(C)c(Cl)c(N)c2)=O)CCC1(F)F CC1(C)CCC(C(N2CCC(NC(C3CC3[N+](=O)[O-])=O)C2(C)C)=O)CC1 C=CCCCCCCC(=O)NCCCOCCN(C(=O)CCN1CCC(F)C1)C c1(C(C)OC(CC2CCC(C)C2)=O)ccc2c(c1)CC(=O)N2 C1(NC(c2ncsc2C)C)C2CCC1CN(C(C1(O)CC1)=O)C2 C1(CNC(C(C)n2cccc2)=O)CCCN(C(c2ccccc2)=O)CC1 N1(C(c2nc(C(C)=O)sc2)=O)CCCC(O)(CNC(C2C(C)C2C)=O)CC1 C1(C(=O)NC2C(C)(C)CN(C(=O)Cc3ccccn3)C2)CCc2ccccc2C1 C1(C)(C(=O)NCC2CC(NC(C(C)Oc3ccccn3)=O)C2)CCCC1O C(CC(CC)C(=O)N(C)CC1CC(F)CN1C(=O)Cc1ccn(C)n1)=CC c1(CN(C)CC2CCN(C(c3cnccc3Cl)=O)CC2)ccc(Cl)cc1 C=C(Cl)CCC(=O)NC(Cc1cc[nH]n1)C(=O)NC(c1ccncc1F)C C1(C(=O)NCC(C#C)CC)CC(C)(C)CN1C(c1ccnnc1)=O N1(C(c2cc(C)sn2)=O)CCC(N(C(=O)CC(C)C(C)(C)C)C)C2(CC2)C1 C(=O)(CC1CCOc2ccccc21)NC(CNC(C(CC(=C)C)OC)=O)CC c1(OC)ccccc1C(O)C(=O)NCC1(C(C)NC(=O)CSc2cnsc2)CC1 c1(CC(=O)NC2CCCC(NC(CC(CN(C)C)O)=O)C2)nc2c([nH]1)CCCC2 N(C(=NCC(C)(C)Oc1ccc(F)cc1F)NCc1ccoc1)CC(C)C c1(C(=O)NCC2CCCN(C(CCCNC(N)=O)=O)CC2)cc2n(c1)CCCC2 N1(C(c2c(C(C)C)n[nH]c2)=O)CC(C(=O)NC2CC(CF)C2)C(C)(C)C1 C(C(C(=O)N1CC=CC(O)C1)C(C)(C)C)NC(C1C(C)CC(=O)CC1)=O CCCC(C)CCCC(=O)NC1CN(C(c2cc3ccncc3s2)=O)CC1(C)C c1(N2CCC(NC(=O)Cn3ccc([N+](=O)[O-])n3)C(F)C2)ncc([N+](=O)[O-])cc1Br C1(NC(=O)CN(C(=O)C(c2cn(C)nc2C)C)CC)CCCCC1CNC(N)=O c1(CC(N2CC(O)(C(C)NC(c3ncccc3F)=O)C2)=O)cccc(O)c1F N1(C(=O)CCc2cccs2)CCCC(C(N2CC3C=CC3C2)=O)C1 C=CC(C)CC(=O)N1CCC(C(=O)NC2CC2CO)(OC)C1 C1(C(C)NC(C2CC(CCO)C2)=O)CN(C(c2cc(C(F)F)cs2)=O)CCO1 C1(CNC(CC(C)c2ccco2)=O)CN(C(c2cc(Cl)cn2C)=O)CC(C)(C)C1 C1(NC(C(CC)n2nccc2C)=O)CC1C1CCN(C(C2(COC)CC2)=O)CC1 N1(C(=O)CCC2CCCO2)CCC2(CCN(C(C3CC4C=CC3C4)=O)C2)C1 N(C(=NCCC(Cl)Cl)NCCF)C1C(OC)OCCC1 N1(C(CNS(N(C)C)(=O)=O)=O)CCCC2(C1)CN(C(C1(C)COCCO1)=O)C2 C(C)(C)(C(=O)N1CCC(CC2CCC2)C1)N(C(CC1(SC)CC1)=O)C c12ccccc1NC(=O)C1C3CN(C1C3)C(=O)N2.c1(SC(C)C)ccccc1I c1(C(N2C3CN(C(C(CCC)N)=O)CC32)=O)ncnc2ccsc12 C1(NC(c2cccc(C(C)C)n2)=O)CC2CN(c3nnc(O)s3)CC2C1 c1(C(=O)NCC(C)NC(C2CCC23CCC3)=O)ccc(-c2ccco2)nc1 C1(C(=O)NCc2n(CCC)ncn2)CN(C(=O)C=CCOCCOC)CC(C)(C)C1 CCCCC(CC)C(=O)N1CCN(C(=O)CNC(=O)NC)CC1CN1CCCC1 C1(O)(CCNC(CCOCCN(C)C)=O)CCN(C(=O)CCC2CCCC2)CC1 S(=O)(=O)(c1ccc(N2CCC(CSC3CC3)C2)cc1Br)NC(CC=C)CO c1(C(N2CCC(CCCNC(c3nc(C)oc3)=O)CC2)=O)ccc(C#N)c(O)c1 C1(CCNC(CCC)(C)c2nnnn2CC2CCOC2)CCCCCC1 c1(C(N2CCCC(N(C(C=CSC)=O)CCO)C2)=O)cc(N(C)C)ccc1F N1(C(C)=O)CCC(C)(C)C1CC(=O)NC1CC(CC(F)(F)F)C1 Cc1ccnc2sc(C(N3CCCOC(CNC(=O)CC(C)C)C3)=O)c(C)c12 Cc1cccc(C(=O)NC2(CO)CCCN(C(=O)C(C(C)O)N(C)C)C2)c1O C1(CCNC(c2c(C)snc2)=O)CCCCN1C(=O)CC1(O)CCC1 C1(CNC(=O)Nc2c(C)nc(C3CCCN(C)C3)o2)CCCC2(CCC2)C1O c1(OC)cncc(C(=O)NC2(C)CC(C(=O)NC3CC(N(C)C)C3)C2)c1 Cc1ccn2cc(CNC(=O)C(=O)Nc3cc(C)c(C)cc3C)nc2c1 c1(C(=O)NC(CCNC(C(c2cnn(C)c2)OC)=O)C)nn[nH]c1C(F)(F)F C1(C(=O)NCCOC2CCN(C(C3(C)CCCC3)=O)C2)CCCC(C2CC2)O1 c1(CC)ccc(NC(C2CC(C)CN2C(c2cc(C)[nH]n2)=O)=O)c(C)n1 C1(C(N(CC=C)CCC)=O)CC(C)N1C(=O)CCNC(=O)CO N1(C(C=Cc2n(CC)ncc2)=O)CCC(CNC(c2cn[nH]c2)=O)C(F)(F)C1 c1(C(=O)NC(CN(C(Cc2ccc(OC)cn2)=O)C)C)c(F)c(N)cc(Cl)c1F C1(C(=O)O)CC(=O)N(C2CCN(C(c3ccccc3CO)=O)CC2)C1 Cc1cccnc1C(=O)NC1CCC(C)(CNC(c2cc(CO)c(C)o2)=O)C1 c1(C(C(=O)OC)N(C)CCNC(=O)Nc2ccc(F)cc2)ccc(C(F)F)cn1 C1(=O)C(CCC)O1.C(=O)(CC(C)=C(C)C)NCCSCCC=C C1(CC)CN(C(=O)CNC(=O)Nc2cc(F)ccc2C)CCN1C(=O)CCCF C=CCC(C)(CC)C(=O)N1CCC(C=CC(=O)NC(C)CC(=O)OC)CC1 n1(CC)cnc(C(=O)NCC(C2CCCC2)NC(=O)Cc2ccccn2)c1 N1(C(CCCc2scc(C)n2)=O)CC2(CCN(C(c3cc(N)ccc3C)=O)C2)C1 C(=O)(C(C)(C)CC(=O)N1CC(O)(CNC(=O)CC(C)(C)C2CC2)C1)OCC C(CCNC(C)=O)(C(C)C)N.C(=O)(C(C)C(C)C)C(C(COC(C)C)NC(C)=O)=O CC1CN(Cc2cccc(Br)c2F)CCS1(=O)=O c1(C(=O)NCC2N(C(C(C3CC3)OC)=O)CC=C2)cc2ncc(Br)cn2n1 N1(C(C2=C(C)OCCS2)=O)CCCC2CN(C(=O)CCC3CCCC3)CCC12 CCC(C)CCC(O)CC(=O)NC(C1CN(c2nc(C(C)C)cc(C)n2)C1)=O CC1CCC(C(F)(F)F)(C(N2CCC2CNC(c2cc(C#N)c[nH]2)=O)=O)C1 c1(OC(C)C)ncccc1C(=O)NCCN(C(c1c[nH]nc1F)=O)C1CC1 c1(C(N2CCC(C(=O)NCc3nc(C4CC4)no3)C2)=O)ccc2c(c1)CCC2 c1(C(=O)NCC2CN(C(C(CSC)O)=O)C(C)(C)C2)ccc2c(c1)CC(C)(C)O2 O=C1CN(CCNC(C2CCC(NC(c3ccc(Cl)cn3)=O)CC2)=O)CCN1 C(=O)(N=c1nc(CC(C)C)s[nH]1)C1CCN(C(C(CC)(C)O)=O)CC1 C#Cc1cc(NC(=O)CC2(CNC(=O)CC(C)CC)CC2)ccc1C N1(C(C2CCC2C(F)(F)F)=O)CCC(O)(c2cn(CC3CC4CC4C3)nn2)CC1 CCC1=C(C(=O)NCCN2CCN(C(=O)C(C3CCCO3)OC)CC2)SCCO1 C#CCCCCC(=O)N(CC(O)CNC(=O)CCc1ccc(SC)cc1)C c1(C(C)C)ccc(C(c2nnnn2C2CC2)Nc2cnc(C(C)OC)s2)cc1 c1(C(N(C)CC2(CNC(=O)Cc3cc[nH]n3)CC2)=O)c[nH]cc1Br c1(OC(c2ccccc2)CC)ccc(CNC(=O)C(=O)Nc2nc(C)cs2)cc1 N1(C(CC2CCC(=O)NC2)=O)CC2(CC2)CC1CC(=O)NCC(=O)NCCO Cc1ccc(C(=O)NCC2CCC2NC(=O)CCCCc2cnn[nH]2)c(N)c1C N1(C(c2c(C(C)=O)scc2)=O)CCCC(CN=[N+]=[N-])C1 CC1(C)CCCC(C(N2CCC3(CC2)CC3CNC(c2cnc(S)[nH]2)=O)=O)CC1 C1(C(N2CC(CC)C(NC(C3(CCOC)CC3)=O)C2)=O)CN2CCC1(C)CC2 Cc1cc(C(N2CC(F)CC2CNC(=O)C=Cc2ccncc2C)=O)cc(N)c1 N1(CCC(=O)N(C(CCNC(C(C)(C)OCCC)=O)C)C)CCCCC1=O c1(C(=O)NC2C(CNC(=O)CN3C(=O)CNC3=O)CCCC2)ccn(O)c(=O)c1 N1(C(=O)CCC2CCCC2)CCC(F)(CNC(C2(F)CC2)=O)CC1 N1(C(c2n(C)c(S)nc2)=O)CC(CNC(C2CC23CCOCC3)=O)CC12CCC2 Cn1cc([N+](=O)[O-])c(C(=O)NCC=CCNC(C2CC2(Cl)CBr)=O)n1 N1(C(C2C(C)(C)OC2(C)C)=O)CC2CC(C1)CN(C(C1CCCO1)=O)C2 N1(C(C(=O)Nc2c(C)nn(C)c2C)C)CCc2[nH]nc(C(F)F)c2C1 O=C(C#CC1CC1)NCc1nocc1C(N1CC(CC(F)F)C1)=O c1(C(N(C2CN(C(c3cc(O)cs3)=O)C2)C)=O)cc2cccnc2nc1O c1(C(=O)Nc2cc(=N)s[nH]2)cccc(-n2cc(C3CC3)nn2)c1.N12CCC(CC1)C2 C(CCC(=O)NC1CC(CCNC(=O)C(C)(C)C2(O)CCC2)C1)=CC Cc1ccc(F)cc1C(=O)NC1C2CCC1N(C(c1cc(Br)oc1C)=O)C2 Cc1ncn(C)c1C(=O)N(CCNC(=O)C(C)C(C)C)C1CC1 c1(C(=O)OCC)nc2c(OC)cccn2c1NC(CCc1ccc(C(=O)OC)[nH]1)=O C1(CNC(CCC(=O)c2ccc[nH]2)=O)CN(C(c2ccc(O)cc2)=O)CC12CC2 c1(C(N2CCC(CNC(C3N(CCC)CCC3)=O)C2)=O)cc(C)cc(Cl)n1 CC1COc2c(C(=O)NC3CCC(CNC(C4(C)CC(F)C4)=O)CC3)cccc21 N1(C(Cc2cc(OC)c(F)cc2)=O)CCCCC2(CCN(C(C34CC3C4)=O)C2)C1 CC(C)CC(O)C(C)C(=O)NCCC(O)C(=O)N(C(CO)C1CC1)C c1(C(C(=O)O)N(C(CCC#C)=O)C2CC2)cccc(Br)c1 N1(CCc2c(OCC)cccc2)CCCOCC12CC2 C1(C(N2C(C(N3CC(CSC)C3)=O)COCC2)=O)CC2(C1)CC2(F)F N1(CSC(C)C(=O)N2CCCC2c2ccncc2)CCOCC1=O.n12cc(nn1)C2 C(C(C)(C)C(=O)N1CCN(CCNC(=O)CC2(C)CCC2)CC1)NC(C)=O C1(C(N2CC(OC)(CO)C2)=O)CCC(C)(C)N(C(=O)Cc2ccsc2C)C1 N1(C(C2(C#C)CCCCC2)=O)CC2CC(NC(C3(C(F)F)CCCC3)=O)CC2C1 c1(C(=O)NC2C(NC(CCN(CCC)C)=O)CCOC2)cc2ccc(C)n2cn1 C1(C(=O)NC2CC(C)(CNC(c3c(C)onc3CO)=O)C2)CN2CCCC2CO1 c1(N2C(C)CCC(NC(c3ccnc4[nH]cnc34)=O)C2)ncc2cc(Br)ccc2n1 c1(CC(=O)NC(C)C(C)NC(C2CCC3(CC2)CC3)=O)c[nH]c2cc(F)ccc12 N1(CC(=O)NCCCC)CC2(CCC(CNC(C3CCN(C)C(C)C3)=O)O2)C1 C(CCCCCF)NC(C(CNC(c1cncs1)=O)N(C)C)=O N1(C(Cc2c(OC)ccc(Cl)c2)=O)CC(NC(=O)C(C)C2CC2)CC12CCC2 CCCCC(CN=c1[nH]cnc2c1COC2)NC(c1nc(C2CC2)ncc1Cl)=O c1(OC)cc(C)c(NC(=O)CC2CN(C(c3nccn3C)=O)CCO2)cn1 c1(C(=O)NC2CC(C)(NC(C(N3CCCC(O)C3)C)=O)C2)ccc(O)c(O)c1 CC(C)(C)CC(O)C(=O)NC1CC(NC(=O)CC2CC3(CCCC3)CO2)C1 c1(C(N(CCCNC(c2ccc(NC3CC3)nc2)=O)C)=O)cc2sccc2cn1 c1(C(=O)OC)ccnc(NC(c2cccc(Cl)c2)Cc2cccc(C)c2)n1 C(N=c1cc[nH]cc1C#N)C1CCCN(C(C(CC=C)(C)C)=O)C1 c1(C(=O)NC2CN(C(CN(C3CC3)CC)=O)C3C2C3)cc2ncccc2s1 C1(CNC(C2C(=O)NCC2)=O)CN(C(C2CC3(CSC3)C2)=O)C2(CCC2)C1 C1(C)(CNC(c2cnc(SC)s2)=O)CCCN(C(=O)CC2CCCCC(=O)N2)C1 C(=O)(CCC(=O)NN(C)C)NC1CCN(C(C(CN(C)C)(C)C)=O)CC1(C)C C1(C)CC(CCN)C1.C1(CC(=O)OC2(C(=O)OCC)CC2)CC(SC)C1 C(C(C)(C)CNC(C1CCCC1CNC(C12CC(C)(C1)C2)=O)=O)OC c1(C(N2CCC(CNC(C(=O)NCC)=O)(CO)CC2)=O)cncc(S(N)(=O)=O)c1 N1(C(c2ccc(C#C)cn2)=O)CCC2(C=C(C(=O)N3CCCC(C)CC3)C2)C1 N1(C(c2cnn[nH]2)=O)CCCC2CN(C(C3CS(=O)(=O)C3)=O)CCC12 C(=O)(CC(O)CC(C)(C)C)N1CCC(C(=O)NCC(CC)O)(CF)C1 c1(CN2CC(C(=O)Nc3ncn(C)n3)C2)ccc(Br)cc1C#N C1(C(N2CC(OC)C(NC(c3n[nH]c(C)c3F)=O)C2)=O)COc2ccccc2C1 C1(CN(C(c2cnc(N(C)C)o2)=O)CC)CCCN1C(C1(CC)CCC1)=O CS(=O)(=O)CCC(=O)N1CCCCC(NC(=O)C(c2ccccn2)O)C1 C(C(=O)N(C1CCCN(C(c2noc(C(C)C)c2C)=O)C1)C)(C(C)(C)C)SC N1(C(c2ccccc2)=O)CCCC(CN2CCCC(Nc3ncc(O)cn3)C2)C1 N1(C(C(C=CC)O)=O)CC(C(=O)NCc2cccc(C)n2)C(CC)C1 CCC(CNC(c1ccccc1)C1CC1)CC(F)(F)F c1(C(=O)NCC2C(NC(=O)C=CC(F)(F)F)CC2)cnc(C(F)(F)F)c(F)c1 CN1C(=O)C(CC(=O)N2CCC3CN(C(C4CC4F)=O)C3C2)c2ccccc21 c1(OC)ccc(C(N(CCC)C(C)C)=O)cn1.C12CCCC1NC(=O)CCO2 C(C1CCCc2c[nH]nc21)NC(=O)CC(C(F)(F)F)n1cccn1 c1(CNC(C2CC(n3cccn3)C2)=O)ncn2c1CCC2 C=CCC(C)(C)C(=O)N1CC(O)(CNC(=O)CCCSC(C)(C)C)C1 C1(NC(C2CCCC(C(=O)OC)C2)=O)CC2CCC1CN(c1nc(C)ns1)C2 CC1CN(C(=O)C(C)(C2CC2)N(C(=O)CC2CSCCO2)C)CCCO1 CN=c1[nH]cc(C(N2CC(CO)(NC(C3CC3(C)C)=O)C2)=O)s1 N1(CC(C)C)CC(C(=O)NCC(C)CN(C)C(c2cc(C(F)F)on2)=O)CC1=O CN1CC(NC(=O)C(CN=[N+]=[N-])NC(C2CC(C3CC3)=NO2)=O)C(F)(F)C1 Cc1cc(C(=O)NCCCC(=O)N(C2CCC2C)C)nc(O)n1 C#CC1(C(=O)NCCC(C)CO)CN(C(c2coc(C)n2)=O)C1 C1(CNC(C(CC)OCC)=O)C(CC)CCN1C(=O)CC(C)(C)C1CC1 c1(C(=O)NCC(C(C)C)NC(C(C=C)O)=O)cnc(C(F)(F)F)c(C)c1 c1(NCC(C(C)C)(C)C)ccc(S(=O)(=O)NCC2CCCOC2)cc1F C1(C(=O)NC(C)COCC2CC2)(CC)CCN(C(=O)C(C)(C)C)CC1 CC#CCC(CO)NC(c1cnn(CCNC(c2ncn(C)n2)=O)c1)=O Cc1ccc(SCC(=O)NC2CCC(NC(C3(C(F)F)CCCC3)=O)CC2)cc1 C(=O)(CC(O)c1ccccc1)N1CC(CN(C(C2(CC=C)CC2)=O)C)C1 c1(CC(=O)NC23CCCN(C(C(CC)O)=O)C2C3)csc2nc(C)cn12 C1(C(=O)NCCC2N(C(C3(C)CCN(C(C)=O)C3)=O)CCC2)CCCCCCC1 Cc1cc(F)c(CN2CCC(CC(=O)Nc3cncc(F)c3I)CC2)c(Br)c1 C1(C(N(C)CCc2cnn(C)c2)=O)CCC2(CC2)N1C(C1C2CCCOC12)=O c1(C(=O)NCC(CNC(c2nnc(O)nc2O)=O)OC)cc2nnn(C)c2s1 c1(C(=O)NCC(C)(C2CC2)NC(=O)CCn2cncn2)cc(C(F)F)nc(Cl)c1 c1(C(N(CC(C)(C)NC(=O)CCP(C)(C)=O)C)=O)nn(C)c2c1CS(=O)(=O)CC2 CC(C)(C#N)C(=O)NCC1CCN(C(c2c[nH]nc2-c2ccccc2)=O)C1 c1(NCC2CC(C)SCC2)nccc(=NCc2ccc(Cl)s2)[nH]1 N1(C(C2(C#C)CC2)=O)C2CCC1(CNC(=O)CSCCN(C)C)CC2 CCCCC(CC)CC(C(=O)Nc1ccccc1Cl)N(CC(C)CO)C CCC(CC(=O)NC1CCC(CNC(=O)CNC(N)=O)CC1)C1CC1 C1(CCNC(c2ccc(CO)o2)=O)(OC)CN(C(C2CC2c2ccnn2C)=O)C1 N1(C(C(C)N(C)C)=O)CCC2(CC1)CN(C(=O)COCc1ncnn1C)CCO2 C(CC(C)(C)C(=O)NCc1ocnc1C(=O)Nc1ccc(F)c(O)c1)SC N1(C(c2ccc(C(N)=O)c(OC)c2)C(=O)NC)CCC(C(=O)OC)=C(F)C1 C1(NC(c2cc(C(=O)OCC)nn2C)=O)CCCCCN(C(=O)C(C)CF)C1 O=C1CC(C(=O)NC2CCC2C(N2CCC23CCC3)=O)=NN1 c1(C(=O)NCC(C(=O)N(C)C)c2ccccc2)ccc2c(c1)CC(=O)N2C c1(C(N2CCCCC(NC(C3C(=O)NCC3)=O)C2)=O)cc2ccccc2[nH]1 C1(CC)CN(C(=O)C(F)C(C)C)CCC1CNC(C1CCCC(=O)N1)=O N1(C(CCCN(C(C)=O)C)=O)CCC(C(=O)N(c2ccccc2C)C)C(C)(C)C1 CC(c1cccs1)=CC(=O)Nc1cccc(NC(c2ccccc2)=O)c1 c1(-c2nc(-c3ccc(OC)cn3)nn2C2CCC(C)C2)ncnc2ccsc12 c1(C(N2CC3C(NC(CCNS(CC)(=O)=O)=O)C3C2)=O)ccc2c(c1)CC(C)O2 Cc1[nH]nc(Cl)c1NC(C1CCN1C(c1cnc(Cl)cn1)=O)=O C1(C(=O)NCC(CC)NC(=O)CCCCCF)CC12CCC(F)(F)CC2 CCCCCC(O)C(=O)N1CCN(C(c2c(CC)nn(C)c2CC)=O)CCC1C S(=O)(=O)(c1cc(C(=O)NCC2(C)CCC(NC(=O)C=CCOC)C2)co1)NC c1(CC)ccc(C(=O)NCC2CCCCN2C(=O)CCN2CCCC2)cc1F N1(C(C2N(C(C)=O)CSC2)=O)CC2CCCC(NC(c3scnc3Cl)=O)C2C1 c1(NC2CCN(C(Cc3ccc(C)cc3)=O)C2)cc(C)nc(CO)n1 CC1CN(C)CC(NC(=O)C(N2CC3CC2CN3C(=O)C(F)(F)F)=O)O1 c1(OC)nc(OC)nc(N2CCC(CCNC(C34CCCN(CC3)C4)=O)CC2)n1 N1(C(C(CCSC)NC(C)=O)=O)CCN(C(=O)CCCC2CCC2)CC(CO)C1 C1(N(C(CCCN(C(C)C)C)=O)C)CC2CC1N(C(c1cncc(N)n1)=O)C2 N1(C(C(C)n2ccnn2)=O)CCOCC1C(=O)N(C1CCN(C)C1=O)C C(=O)(C(F)CCC(C)(C)C)N1CC2C(CNC(CC3CCC(C)CC3)=O)(C2)C1 n1(CCC=C)c(N2CCC(C(F)(F)F)(C(=O)OCC)C2)nnc1C1CC(O)C1 c1(SCCNC(c2cc(Cl)ccc2I)=O)cccc2cc[nH]c12 c1(C(=O)NCCn2cc(CNC(c3n(C)ccc3)=O)nn2)ccccc1CC#N S(=O)(=O)(c1ccc(NC(C2CCCC2)CO)cc1Br)N(C(CCO)c1ccco1)C Cc1nc2[nH]c(C(=O)NCC(C3CCOC3)NC(c3ccccc3)=O)cc2s1 Cc1cc(C)c(C(N2CCC2Cn2cc(Cn3nc(O)ccc3=O)nn2)=O)cc1Br C(=O)(C1=Cc2cc(F)ccc2OC1)N(C)Cc1ccc(Br)cc1 c1(C(N(C(C)C)CCNC(=O)CCC(F)(F)F)=O)ccc2nsnc2c1 Cn1nc(I)cc1NC(=O)NCC1CC(n2ccnc2)C1 Cc1ccc(C)c(C(=O)OCC(c2cn[nH]c2)C)c1 CC(C)C1CNC(=O)COCCO1.c1(CCC(=O)NCCO)nncn1C CC1CN(C(=O)C2=NOCC2)CC1n1cc(-c2ccc(CO)s2)nn1 C1(C(=O)NC(C2CC=CCC2)C(=O)N(CCC)C)CC(=O)NC(=O)N1 c1(CCCNC(N(C)CC2CC2(C)C)=O)cccn1C c1(C(=O)OCC)cccc(=NCC2CC(=O)N(CC3CC3)C2)[nH]1 N1(C(c2c(C)nc(CNC(C3CCCS3)=O)o2)=O)CC(C)(C)CCC1C c1(NC(CC)CCOC)cc(S(=O)(=O)N2CCCOC2)ccc1C#N C1(CC(N2CC(O)(CNC(c3cc(C4CC4)no3)=O)C2)=O)CCCC(C2CC2)O1 C(CN=C(NCC1CCC(=O)N1)NCC1(N2CCOCC2)CCCC1)OC CC#CCC(C(=O)N1CCC1C(C)C)NC(c1c[nH]nc1CC)=O c1(CNC(C(=O)NCc2cccnc2)=O)c(Br)cccc1Br S(=O)(=O)(C(C)CN=c1[nH]c2c(c(=NCCN(C)C(C)C)[nH]1)CCCC2)NC N1(C(CC=CC(C)(C)C)=O)CCCN(C(C2CCCC23CCC3)=O)CC1 c1(C(N(C(C(=O)NC2CN(C(CC)=O)C2)C)CC)=O)cc2cnccc2[nH]1 C1(NC(c2ccnc(N(CCN(C)CC3CC3)C)n2)=O)CCCC(C)(C)O1 C1(CC(=O)N(CCNC(C=CCC)=O)CC)CCCN(C)C1 c1(-c2scc(C(=O)NC3CN(C(=O)Cc4cc[nH]c4)C3)n2)ncccc1Cl c1(C(=O)NCC2N(C(=O)CCN3CCC3)CCC(C)C2)cccc2cccnc12 C1(CNC(CC=CC=C)=O)CC2(CCN(C(c3ccc(C(N)=O)cc3)=O)C2)CO1 c1(CNC(C2CCCC2)=O)ccc2c(c1)CCN(C(c1cccnc1S)=O)C2 C(=O)(C(C)C(C)C)NCC(C)(CNC(c1sc(C)nc1C)=O)OC N1(C(c2cc(CNC(C(n3ccccc3=O)C)=O)on2)=O)CCN(C)CC1CO C(CC(=O)NCC(O)CNC(=O)C(C)c1ncco1)NC(=O)OCC c1(C(=O)NC2COCC2CNC(c2ccncc2F)=O)cc2cc(Cl)ccn2n1 c1(CC)ncc(C(N2CC3CC(NC(=O)Cc4cc(C)no4)C2C3)=O)c(C)n1 C1(CNC(C2C(OCC)C2C)=O)CCN(C(=O)CC2(OC)CC2)CC1 C(=O)(CCCN1CCCC1)NC1CC(NC(CC)=O)C1 C(CC(F)F)(C(=O)N1CC2(CCC2)C1)NC(C(C)(C)n1cncn1)=O C1(CNC(CCc2n(C)cnn2)=O)CN(C(=O)CSCC(N)=O)CC1O C(C(=O)N(C)CC1CCN(C(=O)CCc2ncc[nH]2)C1)(C(C)C)NC(=O)OC CC(C)CCCCCC(=O)N1CC(NC(=O)C(C)OC2CCCCC2)C(F)C1 c1(C(=O)NC2(C)CCN(C(CNC(C(CC)CC)=O)=O)C2)cc[nH]c(=N)c1N Cc1ccc(C(=O)NC2CC(N(C)C(c3cn(C)nc3C(C)C)=O)C2)nc1C c1(C(N(CCC)CCNC(C2CC2C)=O)=O)nccn2c(Br)cnc12 c1(C(=O)NC2CC(F)(CNC(CNC(CC)=O)=O)C2)cc(C#N)ccc1O N1(CC(N2CC(CNC(C34C(CN(C(CC)=O)C3)C4)=O)C2)=O)CCCNS1(=O)=O c1(C(N2CC3(CC(CNC(C(C(C)O)F)=O)C3)C2)=O)ccc2nc[nH]c2c1 c1(CN2C(C)(C(=O)NCC=C)CC2)nc(OC)cc(C)n1 CCCCC(F)(F)C(=O)N1CCC(C2(NC(C34CCC(C3)C4(C)C)=O)CC2)C1 C(CC(=O)N(C)CCc1cc[nH]n1)(CC(C)C)NC(c1c(OC)scc1)=O CCCC(C#N)C(=O)NC(C1CCCC1)CNc1ncc(C(C)(C)O)cn1 c1(C(N2CC3(CN(C(c4c(C)c(O)ccc4)=O)C3)C2)=O)cc2c(ccn2C)[nH]1 C1(COC)C=CCCN1C(=O)C=CC(C)NC(=O)C(C)C1CCC1 c1(C(=O)NC2CCCCN(C(C3CC(C(F)(F)F)C3)=O)C2)cccc2sccc12 c1(C2c3nnnn3N2)c[nH]nc1C.C1(COC)(CC2CC2c2ccco2)COC1 CC(C)C(C(=O)N(CCOCCO)CCO)C(C)NC(C1(C#N)CC1)=O CC(CC#N)C(=O)NC1CCN(CCCNC(=O)CS(C)(=O)=O)C1 C1(NC(C(C2CCC2)OCC)=O)CCCC(C(=O)NCCCS(C)(=O)=O)C1 C(C)(CC(=O)NNC(=O)C(C)(C)CCCCNC(=O)CC1CCCOC1)OC C12(C(=O)NC3C(CC(=O)NC)OCC3)CC(C(=O)OC)(C1)C2(F)F c1(N(C)Cc2c(C)n[nH]c2C)ncnc2c1ncn2C1CCC(C(C)C)CC1 N1(C(C2N(C(CCC=C)=O)CC(N=[N+]=[N-])C2)=O)CC2(CCC2)OCC1C c1(-c2occ(CN(c3c(C)nc(Br)s3)C3CCS(=O)(=O)C3)n2)ccc(F)c(Cl)c1 C(CN=c1[nH]c(=NC(C)c2nc(O)n[nH]2)[nH]c2ccsc12)c1cc(OC)no1 CCC(CC)(CO)C(=O)N1CC(NC(C2(C)C(C)(C)C2(C)C)=O)C(C)C1 C1(C(C)(C)CNC(=O)Cn2ncccc2=O)CCCCN1C(c1cnccn1)=O c1(NC(CCC)CCCNC(=O)C(F)CC2CC2)nccc(C(N)=O)c1[N+](=O)[O-] CC1(C)CC(NC(c2cccc(C3CC3)c2)=O)CN1C(=O)CC1CCCOC1 c1(C(N2CC3C(C2)N3c2ncnc(-c3ccccc3)n2)=O)nc(Cl)ccc1Cl Cc1ccccc1CC(C)Nc1cc(N(C)CCC2CC2)ncn1 c1(CC(N2CCC(CCCNC(CCOCC)=O)C2)=O)c(CC)cccc1CC c1(NCCc2cnc(C)o2)nc[nH]c(=NCc2n[nH]cc2Br)c1C C#Cc1ccc(NC(C2(C)CC(NC(c3cnccc3C)=O)C2)=O)cc1 N1(C(Cc2cncc(C)c2)=O)CC(NC(=O)C(F)C2CCOC2)CC2(CCC2)C1 CN(C)NC(=O)CCC(=O)N1CC2C(NC(c3cccc4oc(O)nc34)=O)C2C1 C1(NC(Cc2cc(C)no2)=O)CC2CC1CN(C(=O)COC(C)C)C2 C1(NC(C=Cc2cc(C)no2)=O)C2CCCN(C(=O)C=CCN(C)C)C2C1(C)C N1(C(=O)CC2CCCC2(F)F)CC23CCCC2(C1)CN(C(C1C2COCC12)=O)C3 Cc1cc(C(=O)N(C)Cc2ccc(NC(C)(C)C)cc2)c2nonc2c1 c1(CC)ccc(C)cc1NC(C1(CNC(=O)CC2(C#N)CC2)CC12CCC2)=O N1(CC)CCCN(C2CC2)CC1.C(CCCC(=O)NCC)N1CCC(C=O)C1 C1(C(=O)NC(c2nc[nH]n2)C)C2CC(O)C(C2)N1C(=O)C(C)CC(F)F N1(C(c2c(N)c(F)ccc2)=O)CC2CC1CCC2NC(=O)CCCS(N)(=O)=O c1(C(=O)NC(c2ccccc2)CC=C)cc(C)cc(I)c1O C(C(F)(F)C(F)(F)CO)NC(N(CC(C)C)Cc1cccs1)=O C1(NC(c2cnn(C(C)C)c2F)=O)CC(NC(C2(C)COC2)=O)C12CCC2 C1(F)(C(=O)NC2CCC(NC(c3nc(COC)sc3)=O)C2)CCS(=O)(=O)C1 C(=O)(CC1=CCCC1)NCCC(=C)CNC(c1cc(F)c[nH]1)=O CC1(C)COCC1CC(N1CCC(NC(=O)C=CC2CC2)C1)=O c1(C(=O)NCCCN(C)C(c2cc(CO)n(C)n2)=O)ccccc1CC(F)(F)F C1(NC(CSC(C)C)=O)CC2CCC(C1)N2C(c1ccc2c(c1)COC2)=O c1(C)ccc(Cl)c2ccccc12.C1(C)(C(C(C2CN(N)CCN2)C)=O)CCOCC1 CC1Cc2c[nH]nc2C(C(=O)N2CC3CCC2C(NC(=O)CN(C)C)C3)C1 Cc1ccc(C(=O)NCCOCCNC(=O)Cc2ccc(O)nc2)cc1 Cc1nn2cc(C(=O)NC(C)(CNC(=O)C(C(C)(C)C)N(C)C)C(C)C)nc2s1 Cc1ccc(C=CC(N2CC(NC(c3cccc(F)c3F)=O)CC(O)C2)=O)cc1 CC(C)C(C)C(=O)NCCC1CC(NC(=O)CCc2ccn(C)n2)C1 N1(C(C23CC(NC(c4ccc(Cl)c(Br)c4)=O)(C2)C3)=O)CC2CCCCC2C1 C12(NC(c3nc(C)nn3C)=O)CCCC1N(C(=O)Cc1cnns1)CCC2 C(=O)(C1CCc2cccc(OC)c21)N(CC(C)NS(CCC)(=O)=O)C CON1CC(NC(C2(C3CCCN3C(=O)CNc3ncccn3)CC2)=O)CC1=O C(=O)(C(C#N)C(C)(C)C)NC1CCC(C(N2CCC(C(C)CO)CC2)=O)CC1 C1(O)(CNC(C=C(COC)C)=O)CCN(C(=O)C(c2cccc(O)c2)C)CC1 C1(OC)CC(CNC(c2ccc(Br)s2)=O)N(C(=O)CNC(C)=O)C1 N1(C(C2(CCC)CC2)=O)CCCC(C2CCN(C(=O)C(O)CCC)CC2)C1 N1(C(c2sc(C)c(C)c2C)=O)CC(C)N(C(=O)Cn2cccc2)CC1C N1(C(CC(CC)C)=O)CCN(C(=O)C(C)(C)OC(C)=O)CC1COC C1(C(=O)OC)CCN(C(CC(C)NCCC(O)COC)=O)CC1 C1(C(N(CC#CC)CC#C)=O)(NC(C2C=C(C)CS2)=O)CCN(C)C1 N1(C(C2CCC3CCC2N3C(C2(CO)CC2)=O)=O)CCC2(CC1)CC2CO CC(C)CC(N)C(=O)N1CCC(Cc2cn(-c3ncccc3Br)nn2)C1 C(=O)(C(C)(C)C(O)C(C)C)NC1C=CCN(C(Cc2cc(OC)cc(Cl)c2)=O)C1 C=C(Cl)CC(C(=O)NC(c1csc(C)n1)C)NC(C1CC(=O)CS1)=O Cc1cc(C(=O)NCC2CCCN(C(=O)CCC3CC3(C)C)C2)c(F)cc1Cl C(=O)(C1=C(Cl)CCCC1)NC1CCN(C(c2ncc(OC)cn2)=O)CC1F C1(NC(CS(N2CCC(C)CC2)(=O)=O)=O)CCC(N=c2ccnc(Cl)[nH]2)CC1 C1(NC(C(c2cccc(C)n2)(F)F)=O)CCN(C(=O)CN2CC3C=CC2C3)C(C)C1 C(N=c1cc(N2CCC(CSc3cccc(Cl)c3)CC2)nc[nH]1)C1(CC#N)CC1 N1(C(CCCCc2cn(C(C)(C)C)nn2)=O)CCNCC(O)C1 N1(C(CSc2n(C)ccn2)=O)CC=CC(CNC(=O)CN2CC3CC3C2)C1 Cc1cc(=NC(C)c2cnsc2)[nH]c(N2CCC(CN3CCCCC3)CC2)n1 C1(OC)CC2CCC1CC2C(=O)N(C)CCN(C)C(C1(C2CCC2)CC1)=O C(C)(CC(=O)NC(C)CNC(=O)C(CC)n1cncn1)N(C(=O)OC(C)(C)C)CC N1(C(CN(C2CC2)CC)=O)CCC(CCNC(C2OCCCO2)=O)C1 C=CCCC(CC(C)C)C(=O)N1CCCC(C(C)Nc2ccccc2[N+](=O)[O-])C1 Cc1cc2cc(C(=O)NC3CC(N(C)C(c4cc(CO)on4)=O)C3)ccc2cn1 c1(CC(=O)NC2(CO)CCCN(C(C(C=CC)O)=O)C2)c[nH]c2c(F)cccc12 C1(Cl)(C(=O)NCC2(CN(C(=O)CN3CCCCC3=O)C)CC2)CC12CCC2 CN1C(=O)COCC1CNC(=O)Cn1cc(CO)nn1 C1(NC(=O)CC2CCCC2)CN(C(c2cc(Cl)nc(Cl)c2)=O)CC2(CCC2)C1 c1(SCC(=O)NCC(CNC(c2n(CC)ncn2)=O)(C)O)ccccc1C S(=O)(=O)(c1cc(C)cnc1NC1CCCCC12CCC2)N(C1CC(SC)C1)C C(=O)(C1=CC2CCC(C1)C2)N1CCC(N(CC(COC)O)C)CC1 C12CCN(C1(C)C)C2=O.C1(N(C)C)CCC(O)(CNC(=O)COC(F)(F)F)CC1 CC(C)CC(F)C(=O)NC1CCC(NC(=O)C(c2ccc(Cl)cc2)C)C1 c1(C(N(C(C)CCNC(=O)Cc2csnn2)C)=O)cnn2c1OCC2 c1(NC(C2COCCN(C(c3c(C)c(CO)ccc3)=O)C2)=O)cc(Br)c(F)cc1F c1(C(=O)NCC(CNC(C(C)Nc2scc(C)n2)=O)O)cc(C)nc(O)n1 C=C(C)CCC(=O)NC(C1CCCN1C(c1ccc(C2CC2)o1)=O)C c1(OC)ccc(S(=O)(=O)NCc2cc(C#N)n(C)c2C)nc1 CCC(F)(F)C(=O)N(C(C)CCNC(c1cn(-c2cnn(C)c2)cn1)=O)C N1(C(CC(CC)O)=O)CCC(C2(O)CN(C(=O)C=CC3CCOC3)C2)CC1 Cc1ccc(OCC(N2CC(CC(C)NC(C3CC(O)C3)=O)C2)=O)c(F)c1 CC1(C)CC(CC(N2CC(CC(N)=O)C2)=O)CN1C(=O)CCSc1cn[nH]c1 C(=O)(C(CO)C(C)(C)C)NCc1nc(C)c(C(N2CCC2C(=O)N(C)C)=O)o1 C1(C#CC(=O)NC2CCCC(NC(=O)C=C(C)C(C)(C)C)C2)(CC)CC1 Cc1ccc(C(=O)NCCCN(C)C(c2cnc(O)c(Cl)c2)=O)cc1Cl N1(C(=O)Cn2cnnc2)CC(S(=O)(=O)N2CCN(C(=O)C(O)C3CC3)CC2)C1 C1(c2ccc(Cl)cc2)(C(C2CC2n2cccn2)=O)CCCC2(CCC2)C1 C12CCC(=O)N(C1)CC2=O.c1(CC)csc(CC)n1.C(CN(C)CCN)OC1CC1 C1(CCNC(C(CC2CCC2)NC(C)=O)=O)CSCCN1C(c1cncs1)=O C1(NC(N2CC(C)C(c3c(F)cccc3F)C2)=O)CCCN(C)CC1 c1(CNC(=O)OC(C)(C)C)cc(C(=O)Nc2cnoc2)ccn1 C(=O)(C(C)CC(C)(C)C)NC1(C(N2CC(CC)OCCC2)=O)CCN(C)C1 c1(OC)ccc(C(=O)NC(C)CC(C)NC(c2conc2C)=O)c2ccncc12 CCCCCCC(=O)N1CCC(N(C)C(c2ccc(N)c(OC)c2)=O)C1 CCCCC(CC)C(=O)N1CCSCC1CCNC(=O)C=CCN(CC)CC CC1(C)CC(C(N2CCC3C(NC(c4c[nH]c(=N)s4)=O)C23)=O)CCO1 C1(NC(C2CC(=O)NC2)=O)CCCN(C(=O)CCc2nnc(C(F)F)o2)CC1 C=CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cccnc3OC)=O)C2)CC1 c1(C(=O)NCC2CCN(C(CCSc3n(C)nnn3)=O)C2)ccccc1CC#N N1(C(c2c(SC)scc2)=O)CCC(C)(CNC(C2C3CCCCC23)=O)C1 c1(OCC)nc(Cl)ccc1C(N1CC2(CC(NC(=O)CCSC)C2)C1)=O Cc1ccc2c(c1)CCC2NC(=O)CCCc1cccs1 CC1CCCN(C(c2cnc(C3CC3)nc2)=O)C1NC1CC1.C12CC(C1)NC2=O N1(C(CS(=O)(=O)N(C)C)=O)CC(C2CN(C(C3CCC(C(F)(F)F)C3)=O)C2)C1 N1(C(CC(CC)SC)=O)CCCCCC(NC(c2c(N)nn3ccccc23)=O)C1 C1(NC(c2cc(-c3cccnc3)[nH]n2)=O)CCN(C(C2CC2C2CC2)=O)C12CC2 C1(C(=O)NC2CCCN(C(=O)Cc3c(F)cccc3F)C2)CCC2C(C1)C2(F)F c1(OCC)ccc(Cl)cc1CN(C(=O)NC(C)C(C)C)C1CC1 C(=O)(CC1OC(=O)Nc2ccccc21)NCC(CNC(Cn1ncc(C)c1)=O)O C1(CC(=O)NC(CNC(C(CCC)C(C)C)=O)(C)C)C2CC3CC(C2)CC1C3 C(=O)(CCC(CC)NC(C1CC2CCC2C1)=O)NCCSCCC=C C(C)(CCC(=O)NCC1(F)CCN(C(=O)C=CCn2cncn2)C1)OC N1(C(C2CC(N3CCC3)C2)=O)CCC(CN(C(C2CCC2)=O)C2CC2)CC1 c1(CCC(=O)OC)ccc(C(=O)NCC(C)CNC(C2(C)CCOCC2)=O)cc1 O=C(CCC(=O)c1cccc(Cl)c1)NCC(CO)NC(C1CCCC12CC2)=O C(c1cccc(F)c1Cl)=CC(=O)NCC1(NC(C2C(OC)(OC)CC2)=O)CCC1 N1(C(CN2C(=O)C(C)C(C)C2=O)=O)CCC2CCN(C(C3(CO)CC3)=O)CC12 C1(NC(CN(C(C(C)N(C)C)=O)C)=O)CCC(O)C(O)C1 C1(COC)(CNC(C2(C)CCOC2)=O)CCN(C(=O)CCCSc2ccccc2)C1 N1(C(C2(O)C(C)(C)C2)=O)CC(CO)C2(C1)CN(C(c1cc(F)ccc1Cl)=O)C2 CC(C)(C)C(CCO)C(c1ccc(=O)n(Cc2cccc(F)c2)n1)=O O=C(CC1=CCCCC1)NC1(C(=O)NCC2(C3CCC3)CC2)CC(F)C1 N#Cc1cccc(NC(c2sccc2CNC(C23CC(CO)(C2)C3)=O)=O)c1 S1(=O)(=O)c2ccc(c(Cl)c2)NCC2(CCC2)N1C.C1(N)CC(CO)C1.CO C12CC3CC(C3C1)C(=O)N2.c1(C2CC(=O)C2)ccc(C(F)(F)F)o1.C(=O)C(F)=C(C)C C1(OC)CCC2(C(=O)NCC3CCCC(CNC(c4cccnc4C)=O)C3)CC12 c1(CC)ncc(C(N2CC3C(C(=O)Nc4cnsc4)C3C2)=O)cn1 C(CCNC1CC1)(C(=O)N1CCCC2CC12)N.O=CCCOCC1CCC1 C(=O)(C1=CC(C)(C)C1)N1CC(SC)C(C(=O)NCC2(CC(C)C)CC2)C1 Nc1ccc(C(=O)NC2CN(C(=O)CC3CCC(C(F)F)O3)C2)c2cnccc12 c1(C(c2nnnn2CCNC2CCC2)Nc2nc[nH]n2)csc(C2CCCO2)n1 Cc1cc(C(=O)NCC2CC2CNC(=O)C(C)(C)c2ccc(Cl)s2)c(C)cc1Cl N1(C(C2(C)C(C)CCC2)=O)CC(NC(c2coc(C(F)F)n2)=O)C(C)(C)C1 Cc1sc2ncc(C(=O)NC(C)CN(C)C(C3CC34CCOC4)=O)n2c1C CN1CCN(C(=O)CCN(CCO)C(C2CCC(C3CC3)C2)=O)CC(O)C1 CC1CN(C(c2ccno2)=O)CCC1NC(=O)CC1CCC(=O)C1 c1cc2[nH]c(=NC3CN(NC4CSCCO4)C3)[nH]c(=NC3CC3)c2s1 c1(OCC(=O)NCCCC(C)NC(C2(C#C)CC2)=O)ccc(C(F)(F)F)cn1 CC(CC(C)(C)C)C(=O)NCC(C)(C)C(N1C2CCC1CC(O)C2)=O c1(CCC(N2CC(NC(C(C)OC)=O)C2)=O)ccccc1N=[N+]=[N-] c1(C(N2CCC(CNC(c3cnc(C)[nH]3)=O)CC2C)=O)cccc2oc(=N)[nH]c12 N1(C(=O)NC(C#C)(C)C)CCC2(CC1)CC2NC(N1CCC(C(N)=O)CC1)=O c1(C(=O)NCc2occ(C(=O)NCC(COC)O)c2)nccc(C)c1F C(=O)(N1CC(C)(O)CO1)c1ccc(CNC(N2CCCC(C)C2)=O)cc1 CC1(F)CCC(C(=O)NC2CN(C(=O)CN3CC=CC3)C(C)(C)C2)CC1 C(=O)(C(C(C)(C)C)OC)N(C1CCCN(C(c2n(CC=C)ccc2)=O)C1)C CC(C)(C)C(C(=O)N1CCC1CNC(C1CC1C(F)(F)F)=O)c1cc[nH]n1 C1(NC(C(C)OCC)=O)CN(C(c2cnn(C)c2SC)=O)CCC1(C)C C1(O)(CCNC(C(C)NC(c2ccc(Cl)cc2Cl)=O)=O)Cc2ccccc2C1 C1(NC(c2c(C)nn(C)n2)=O)CN(C(c2ccnn2C(C)C)=O)C2CCCC12 C1(NC(C(C2CCOCC2)C)=O)CC2CCC(C1)N2C(c1cc2sccc2s1)=O c1(C(=O)NCCN(C(c2c(C)nc(C(C)C)s2)=O)C2CC2)cnn2c1CCC2 N1(C(c2c(COC)onc2)=O)CCC(C(=O)NCC(C)S(N)(=O)=O)CC1 N1(C(c2cn3ccsc3n2)=O)CC2CCC(C1)N2C(c1cc(F)c(O)c(F)c1)=O CCCCC(O)C(C)C(=O)N1CCC(C(=O)NCCc2ccc(O)cn2)C12CC2 CCC(CC)(C(=O)NC1CCN(C(=O)CC2=CCOCC2)CC1)C(C)C C1(CCC)CN(C(=O)C=CC2CC2)CCN1C(=O)C(CC=CC)c1ccccc1 C1(NC(=O)C=C(Cl)Cl)CCN(C(c2ccc(-c3cc[nH]n3)nc2)=O)CC12CCC2 O=C(CCCc1cncs1)NC(C1CCOC1)(C1CC1)C1CC1 C#Cc1ccccc1CC(=O)NC1CCC(NC(c2cn(C(C)C)nc2C)=O)C1 N1(C(C(=O)NCCC)C(C)C2CCOC2)Cc2ccccc2CC1CC c1(C(C(=O)NCCOCC)N(C)CC)csc(Br)c1.C12(N)CC(C1)C2 N1(C(Cn2nc(C)oc2=O)=O)CC(NC(=O)C=CC(C)C)CC(F)C1 c1(CNC(C2C(OC(C)C)C2)=O)cccnc1C(F)(F)F N1(CCn2c(=O)cc(CC(=O)OCC)[nH]2)CCC(c2nn[nH]n2)(SCC)CC1 C(=O)(C(C)(C)CC(C)(C)C)NCCCCC1CCCN(C(c2ncn(C)n2)=O)C1 N1(C(c2n[nH]c(C)c2F)=O)CC(CNC(c2ccc(F)cn2)=O)C(C)(C)C1 C1(C(=O)NCCC(C)NC(=O)C2=CCCSCC2)CC12CC(F)(F)C2 C1(NC(CCCN(C(=O)CC2CC(=O)NC2=O)C)=O)CC2(CCCCO2)C1 CC(C)CC(CN1CCCC1)NC(=O)C(C1CC1)NC(c1ccccc1)=O c1(CC)nccc(C(=O)NC2CC2CNC(C2(CCCC3CC3)CCCC2)=O)n1 Cc1cc(=O)c(C(=O)NC(C)CC(C)NC(C23CCCC2(C(N)=O)C3)=O)cn1C CCCCCCn1nnnc1CN1CCCC1c1cc(C(=O)OCC)co1 C1(CNC(C(C2CCCOC2)OC)=O)CCN(C(c2nccnc2CO)=O)CC1 c1(C(CNC(CC2(C(=O)NC3CC3)CCC2)=O)NC(=O)NC)ccncc1.OC C1(C(C)CO)CCN(C(C2CCCC2NC(C2CC2c2ccccc2)=O)=O)CC1 N1(C(C(CCC(C)C)NC(Cc2c(C)cccc2)=O)=O)CCc2ccccc2C1 CC1(C)CCCN(C(c2ccc(=O)n(C)c2)=O)C1C(N1CCC2(CSC2)C1)=O CN1CCN(C(C2CC(F)CN2C(C2(C#N)CC3CC3C2)=O)=O)CC1CO C(c1c(Cl)nc2ccccn12)=CC(=O)NC1CN(C(CC2(C)CCC2)=O)CC1O c1(C(N(CC(C)CNC(C2CCCC(C)(C)C2)=O)C)=O)cc2c(nn1)CCC2 C(=O)(C(C)C(O)CC(C)C)N1CCC(CC)C1C(N1CC2(CCC1CO)CC2)=O N1(CC(=O)OCc2c(C(=O)OCC)scn2)CCC(CN)CC1 CC(N=c1[nH]c(=NCC2CCS(=O)(=O)C2)[nH]c2ccsc12)c1ncc[nH]1 C1(C)(C(N(C)CC2CCN(C(C=C3CCC(C)C3)=O)CC2)=O)CCCCNC1=O Cc1ncc(CCC(=O)N(c2ccccn2)C(N2CCCCC2)=O)c(O)n1 CC1(CNC(c2c[nH]cc(Cl)c2=O)=O)Cc2ccccc21 C(=O)(C(C)(C)CCS(C)(=O)=O)NCC(CO)NC(CSC)=O c1(OCC(=O)NCCCN(C(CCCC)=O)CC)ccnc(C(F)(F)F)c1 Cn1nnc(C(=O)NC2CCC2CNC(c2cc[n+]([O-])cc2)=O)c1C(F)F n1(CC)cc(C(=O)NC(C)(C)CCCNC(=O)CCC(C)SC)c(C(C)(C)C)n1 c1(COC)ccccc1C(=O)NC(C)(CNC(c1sccc1CO)=O)C1CCC1 c1(C(c2nnnn2CCOCC)NCC=CC)c(C)noc1CC c1(C(=O)NCCCCNC(Cn2nnc(C)n2)=O)ccc(O)nc1Cl c1(NC(CSCCC(N2C(C)(C3CCC3)CCC2)=O)=O)cc(F)ccc1O c1(Nc2cccc(C(=O)NS(C)(=O)=O)c2)cncc(F)c1Br C1(NC(C(CCC)NC(=O)C(C)=C2CC2)=O)CCOC2(CCC2)C1 c1(C(N2CC3(CN(C(CN4C(C)CCCC4C)=O)C3)C2)=O)ccc(Cl)c(C#N)n1 c1(C(N2CC(C)(NC(C(CC)SC)=O)C2)=O)cnc(O)n(-c2ccccc2)c1=O C=CCCC(C)(C)C(=O)NCCCCC(C)(C)C.C12CSCCN1C2=O C#Cc1c[nH]nc1C(=O)NCC=CCC(=O)NC(CN(C)C)CC(C)C c1(C2(C#N)CC2)ccccc1C(=O)NC1CCCCC1NC(C1CCCCS1)=O N1(NC(N2CCC(C3CCC(F)(F)CC3)C2)=O)CC23CCCC2(C1)CS(=O)(=O)C3 C1(C(=O)NCCc2cncn2C2CC2)CCCCC1C1CC1 c1(C(N2CC(O)(CNC(C(C)SC)=O)C2)=O)cc(N)c(C(=O)NC2CC2)s1 Cc1ccc2cccc(CNCc3c(Cl)cccc3Cl)c2c1 C1(CN(C)C)CN(CC)CCN1Cc1ccc(=O)n(-c2ccc(F)cc2)c1 N1(C(c2c(C)[nH]nc2Cl)=O)C2CCC1CC(N(C(=O)CN1CCCC1C)C)C2 Cc1cc(C(=O)NC2CCCC2C(=O)Nc2ncc(Br)nc2C)c(C)cc1Br CC1CN(C(=O)CN2CCCNS2(=O)=O)CCC1NC(=O)C(C)(C)NC(N)=O CC1OCCC1(C)C(N1CC(O)(CCNC(c2cnn(C)c2Br)=O)C1)=O C(=O)(C(CC)C(=O)N1CCN(C(C2(COC)CC=CCC2)=O)CC1)OCC c1(C(=O)NCCNC(C2C(CC)CCC2)=O)cccc(OC)c1[N+](=O)[O-] N1(C(c2nc(C)sc2)=O)CCC2C(CCCN2C(=O)COCC2CCC2)C1 C(C(C)(C)C(=O)NC1CC1NC(=O)Cc1coc(C(F)F)n1)OC(C)C C1(NC(c2cc(CC)[nH]n2)=O)C2CC1N(C(=O)C(C)Oc1ccc(Cl)cc1Cl)C2C N1(C(C(C(CC)C)C)=O)CCN(C(=O)C(C)N(C)C)C2COCC12 C1(C(=O)NC(CN(C(c2n(CCC)ncc2)=O)C)C)Cc2cccc(F)c2O1 c1(OC)c(C)cc(C(=O)NC2CCN(S(=O)(=O)c3cccnc3)CC2F)cc1C N1(C(COCC(C)C)=O)CCOC(C(=O)NCc2ncc[nH]2)C1 CC1CN(C(C2(Oc3ccccc3)CC2)=O)CC1CNC(C1(CCC)CC1)=O Cc1cc(CNC(=O)CCC2CCCCN(C(=O)C3=C(Cl)CCC3)C2)cc(F)c1 C1(N(C(=O)CC(F)F)CC(C)C)CCN(C(c2csc(-c3cn[nH]c3)n2)=O)CC1 Cc1cc(F)c(C(N2CC(c3cn(CSC4CC4)nn3)C(O)C2)=O)cc1Cl c1(C(=O)NC(C)C(C)NC(c2cscc2C(N)=O)=O)nnn2c1C(=O)NCC2 N1(C(C(F)=CCC)=O)CC2CCOC2(CNC(=O)C(C)CC(N)=O)C1 N1(OC(CCCC#C)=O)CCN(C(=O)CCCc2ccc(C(C)(C)C)cc2)C2CC12 CC1COCCC1CNC(c1ccc(CNC(C2C3CC4C(C3)C24)=O)s1)=O N1(C2CCCC2)CC(NC(C2(C(=O)OCC)CC2(F)F)=O)CC(O)C1.CCOCC N1(C(c2c(C)oc(C(C)C)n2)=O)CCN(C(=O)CC2CCCCC2O)C(CO)C1 c1(OCC)cccc(-c2cn(CCNC(=O)C(C)c3cc[nH]n3)nn2)c1 C=CC(O)C(=O)N(CCNC(=O)Cc1cnc(C)s1)CCc1ccccc1 c1(OCCC(N2CC(OCCNC(=O)C=Cc3ccco3)C2)=O)ccccc1F C1(C(=O)NC2CC3CC(NC(c4cccnc4)=O)CC32)CN=C2N=CNN2C1 S(=O)(=O)(c1csc(C(=O)NC2CC(O)CN(C(=O)Cn3ncnn3)C2)c1)NC C1(SC)CC2C=CC1C2.N12CCC(CC1)C1CCC(C1)C2=O N1(C(CCN(CCC)C)=O)CCC(C)N(C(C23CCC(OC)C2CC3)=O)CC1 n1(CC)ccc(C(c2nnnn2CCC2(C)CC2)NCc2ccsc2C)n1 C(=O)(CCC1CCC1)NC1(C=O)CSC1.c1(C2N(C(C)C3CC3)CC2)cnc[nH]1 c1(CC)nc(C)c(C(=O)NC2CC(CNC(c3coc(C(C)=O)c3)=O)C2(C)C)o1 Cc1nnc2n1CCC2(C)C(=O)N(CCCCCNC(c1cccc(Cl)c1)=O)C Cc1cc(CNC(c2ccnc(O)c2)=O)oc1C(=O)NCc1cnn(C)c1O N1(Cc2ccc(CC)s2)CC2CCC1CN(C(=O)CN1CCN(C)C1=O)C2 CCC(C)CCCCC(=O)N1CCC(NC(c2cccn(C)c2=O)=O)C(C)(C)C1 C(=O)(N=c1nc(C2CCOCC2)[nH]s1)NC(C)CNC(=O)Cn1cncn1 CCC(CNC(c1cc(CNC(=O)Cc2cc(C)n(C)n2)ccn1)=O)C(C)C c1(-c2ccc(C(=O)NCC(C)NC(=O)CNC(N)=O)s2)ccccc1F C(=O)(C(CC(C)CC)NC(C1CC2(CCC2)CO1)=O)NCc1cnc(CC)[nH]1 c1(NCC(=O)NCC2(C)CCN(C(c3cscn3)=O)C2)ccc(F)cc1F c1(OC)coc(C(=O)NCC2CC(C)(C)CN2C(=O)CN2CC3CC3C2)cc1=O c1(C(=O)NCC(C)NC(C2CN(C)CC2C(F)(F)F)=O)noc2cc(Cl)ccc12 C1(CC(=O)NC(CNC(c2ncc(OC)nc2)=O)(C)C2CC2)CCOC(C)(C)C1 c12ccc(cc1F)[nH]2.C1(COC)CC2CC2C1=O C1(C(N2CC(CN(C(c3cc(OC)n(C)n3)=O)C)C2)=O)CC12CCOCC2 N1(C(c2c(C)oc(C(C)C)n2)=O)C2CCCC1CC(NC(C1CC(CF)C1)=O)C2 C=CCCN=C(NCCc1ccc(C)nc1OC)NCC1CC(C(F)F)C1 C12(C(=O)O)CCC(=O)C(N3CCOCC3)CCC1C2.N#Cc1ccc2c(c1)N2 CCC(Cc1ccccc1)C(=O)NC1CN(C(C2CC(N(C)C)C2)=O)CC1OC CC1(C)CC=C(C(=O)N2CCC(OCCNC(C3CC4(CCCO4)C3)=O)C2)CC1 c1(OC)ccc(Br)c(S(=O)(=O)N2Cc3cnn(-c4ccc(Cl)cc4)c3C2)c1 N1(C(C2N(C(CCC)=O)CSC2)=O)CC2C(NC(=O)C3=CCOC3)C2C1 c1(CNC(C(c2ncc[nH]2)C)=O)nocc1C(=O)NCC(C)N(C)C1CC1 C(CN=c1nc(N2CCC(C)(F)CC2)cc[nH]1)C1(CC)CCCCC1 C1(NC(C2CC2(c2ccccc2)F)=O)CCN(C(c2cn[nH]c2)=O)C1 CC1CCc2[nH]nc(C(=O)NC3C=CCN(C(=O)CC4COC(=O)N4)C3)c2C1 C1(C(=O)NC(C2(O)CN(C(c3nc(C)c(C)s3)=O)C2)C)CCOC2(CCC2)C1 c1(N(C)CC2CCN(C(=O)C=Cc3cscn3)C2)cc(C(C)(C)C)nc(Cl)n1 CC(C)CC(CNC(C1CCS1(=O)=O)=O)NC(=O)CC1(C(F)F)CC1 N1(C(C(F)=CC)=O)CCN(C(=O)CCN2C(C)CCCC2C)CC(C)(C)C1 Cn1[nH]c(=NC(=O)C2CCN(C(C3CC(=C4CCC4)C3)=O)CC2O)cc1C1CC1 c1(SCCNC(CNC(C(c2ccccc2)C)=O)=O)ccccc1Cl c1(OC)ccc(CN2CCC(F)(CNC(c3cc(O)no3)=O)CC2)cc1C(C)C C1(NC(C=C(COC)C)=O)CCCCC1CO.C12(CCCCC1)C(F)(F)C(=O)N2 C1(C2CN(C(c3scnc3C)=O)C2)(NC(c2cn(CCOC)nn2)=O)CC1 N1(C(COC2CN(C(C3(C)CC4(CCC4)C3)=O)C2)=O)CCC2(CCC2)CC1 C(C(CNC(=O)CCSC1CCCC1)C(F)(F)F)NC(C1OCCC(C)C1)=O N1(C(Cc2cc(C)sc2)=O)CC2(C=C(C(=O)NCC(C3CCCC3)O)CO2)C1 C12(C(N(C(C)C(F)F)C)=O)CC3CC(CC(C3)C1N)C2 CCC(CC)(CO)C(=O)NC1COC2(C1)CN(C(=O)CCC(=O)N(C)C)C2 C1(CNC(C(C)OCCOC)=O)CCC(C(=O)NCCC(O)C2CC2)C1 c1(C(C2CCC(O)C2)C(=O)NCC2(NC(=O)C=CCBr)COC2)ccc(F)cc1 N1(C(C(CCC)C(C)C)=O)Cc2n[nH]cc2C1C(=O)N(C)CC1CC1C c1(C(=O)NC23C(CCN(C(CCC#CC)=O)CC2)C3)ccc2nn(C)cc2c1 C(=O)(CC1=CCCCC1)NC(CCOC)C(N1C2CCC1C(COC)C2)=O C1(NC(c2cc(C(C)=O)sc2)=O)COC2(C1)CN(C(=O)CC1CCCO1)C2 C12(C(=O)NC3CN(C(c4csc(Cl)n4)=O)C3)CCCC1CC2 C(=O)(CCCNC(=O)C(C)CNC(c1csc(F)c1)=O)OCC C#CCC(O)C(=O)N(C1CCN(C(c2cnn(-c3ncc(Cl)cn3)c2)=O)C1)C C#Cc1cccc(CCC(=O)NCc2ccccc2C)c1.C1(=O)C=CC=CCN1 O=C(C1COc2ccccc21)NCC1CC(O)CN1C(c1cccc(CO)n1)=O c1(OCC)cccc(C(=O)NC(C)(C)CCCNC(=O)CCC2CC2C)c1N C(=O)(CCCC(C)(C)CC)NC1CC2CN(C(C3(CCCC)CC3)=O)CC2C1 N1(C(CSCCCC)=O)CC2C(C(=O)N(CC)CC3CCOC3)C2C1 CCC1=NOC(CC(N2CCCCCC2)=O)C1.N12CCC(C1)OCC2=O CC(O)CCCCCC(=O)Nc1ncc(Cc2ccccc2)s1 N1(C=O)CC2CCN(C(=O)CCN3CCC(O)CC3)CC2C1.c1(CC)cscn1 c1(NC(C2CCCN(C3CCC3)C2)C)ccc(S(N)(=O)=O)s1 c1(OC)ccc2c(=NCc3nnc4n3CCS4)[nH]c(=NC3CC(C#N)C3)[nH]c2c1 c1(CC(=O)OC(C(=O)NCC=C)C)ccc(C)c(C)c1 N1(C(c2nnn(C)n2)=O)CCC2CCN(C(C3(O)CCC3)=O)CC12 CCCCCC(O)C(=O)NCCCN(C)C(c1cn(-c2ccc(Cl)cc2)nn1)=O N1(C(C2C(OCc3cc(-c4ccccc4)nn3C)C2)=O)CC2CCC1CN2CC C=C(C)C(CC(=O)NCCCNC(=O)CC1CC2CC2C1)OCC c1(C(N2CCC(CNC(C(CC(N)=O)O)=O)C(O)C2)=O)cc(Cl)cc2c1CCC2 C1(C2CCCN(C(C3(CF)CCC3)=O)C2)(NC(c2cc(C)c(=O)n(C)c2)=O)CC1 C12(CNC(C=CC=CCC)=O)CCCC1N(C(c1nnc(CC)s1)=O)CCC2 C1(NC(C2(C)CC=CC2)=O)CCCCC1CC(=O)N(C)C.C1(C)(C)C(=O)N1 c1(CNC(C=CC)=O)ccc(CN(C(C(=O)NCC)CC)C)cc1 C(CCS(=O)(=O)C(C)(C)C)N(CC(CCCCCC)CC)C1CC1 c1(OC)ccccc1C(C)=CC(=O)NC(C)CCN(C)C(C1(F)CC1)=O C(=O)(C(C)CC(C)C)NC(c1cccc(OC)c1)CNC(C1(C)CCC(=O)C1)=O CC(C)C(O)C(C)C(=O)N1CC2(CC(CC(N3CCCC(C)(C)C3)=O)C2)C1 C1(NC(C=CCOC)=O)CCN(C(c2ccc3c(c2)OCO3)=O)CC(C)(C)C1 C=CCCCC(C)(C)C(=O)NCC1CN(C(=O)CCc2nccn2C)C2CC12 N1(C(C(C)OCCS(=O)(=O)NC2CCC2)=O)CC(=O)CC1C(=O)NCC1CC1 Cc1ccc(C(=O)NCCC2CN(C(c3ccsc3C(F)F)=O)CCO2)c(O)c1 c1(CN2C(CC(=O)NC(C)C)C(=O)NCC2)cnc2ccccc2c1 c1(OC)cccc(C)c1C(N1CCC(CN(C(=O)C#CC2CC2)C)CC1)=O C1(CNC(C(C)N(C)C)=O)C=CCN1C(c1cnc(CC(C)(C)C)o1)=O C12(NC(COCC)=O)CCOCC1CN(C(=O)CCc1ccc(Br)cn1)C2 C(=O)(C(O)C(F)(F)F)N(CCC)CC1N(C(CC2(CC(=O)OC)CC2)=O)CCC1 C(=O)(C1=CCN(C(c2cnc(Cl)n2C)=O)C1)NC(C)Cc1ccccc1 C(=O)(C1=CCCC(C)(C)C1)N(C)CC1N(C(C(C(C)C)CO)=O)CCOC1 CCCS(=O)(=O)CC(=O)N(C1CCCN(C(c2ccc3oncc3c2)=O)C1)C CC1(C)CCOC(C(N2CCN(C(=O)COCc3nc[nH]n3)CC2CO)=O)C1 C(CCS(C)=O)(C(=O)NCCc1cc(O)c(O)c(O)c1)N(C)C C=CCC(C(=O)N1CCN(c2nc3ccccc3o2)C(CCCC)C1)C(C)C N1(C(C(CC(C)C)ONC(=O)C(F)N(C)C)=O)CC2(CCC2(C)C)C1 N1(C(C2CC(CN(C)C)C2)=O)CCCC1CCNC(=O)C(F)C1CCOC1 c1(C(=O)NC(c2ccccc2)C2CC2)cnn(Cc2ccccc2)c1Cl C1(CNC(C2(OC)CCN(C(C3CCC4(CC4)C3)=O)C2)=O)CC2(C1)CC(O)C2 c1(OCCCC(=O)NC(CC)CN(C)C(C2(F)CC2)=O)ccc(Cl)cc1C C1(C2CCCO2)(c2onc(CC(C)C)n2)CCCO1.c12ccnc(c1)S2 CCC(C)(COC)C(=O)N1CCC(CC(C)NC(c2cnnc(O)c2)=O)CC1 S(=O)(=O)(c1c[nH]c(C(=O)NCC2CCCCN(C(c3ccc(C)o3)=O)C2)c1)NC c1(C(=O)NCC(CNC(=O)C(C2(O)CCCC2)F)OC)snnc1C1CC1 n1(CC(=O)N(C2CN(C(=O)COc3cncc(Cl)c3)C2)C)cnc2ccccc12 C1(CNC(C)=O)CN(C(=O)C=Cc2ccnn2CC)CC2(CCC2)O1 C1(C)(NC(=O)CC(O)C2CCCC2)CC1(C)C.CC1(C)C=CC(=O)N2CC1C2 C1(NC(Cn2cc(N)nn2)=O)CN(C(C2CC(C(=O)OC)C2)=O)CC12CCC2.OC c1(OCC)cccc(C(=O)NC2CCC(NC(C3CCN(C)C3=O)=O)CC2)c1 N1(C(COCCC)=O)CCC2(CCCC2NC(C2CC3C=CC2C3)=O)CC1 C1(C)(CNC(c2c(COC)ccs2)=O)CN(C(c2ccccc2C)=O)CCO1 C1(CC(=O)NC2CC(NC(c3n(C)c(=O)ccc3)=O)C2)CSc2ccccc2O1 c1(C(N(CC(=O)NCc2cc(F)ccc2F)CCOC)=O)ccnc(O)c1F C1(CN(C)C(C2C(C)(C)C2(C)C)=O)CN(C(c2cnc(N(C)C)s2)=O)CCO1 CC1(O)CC2(CN(C(=O)C(c3ccc(C4CCCCC4)cc3)=O)C2)C1 c1(CNCCN(CCOC)C(c2occc2C)=O)cc2ccc(OC)cc2cn1 N1(C(C(c2cncnc2)C)=O)CCCC1(C)CCC(=O)NC1(CN(C)C)CC1 CN1C2CCC1CC(C(=O)NCCCNC(c1cnc3n1CCCC3)=O)C2 c1(C(N(C2CCC(NC(C=CC)=O)CC2)C)=O)nc(OC)ccc1F C(C(F)(F)C(F)(F)CO)NC(=O)NC(c1nnc(CNC(C)=O)s1)C C(=O)(C(CC(C)C)N(C)C(C1CC(C(C)C)=NO1)=O)NCC(C#C)OC c1(C(=O)NC2CC(NC(C3(N(C)C)CCC3)=O)C2)ccncc1NSC c1(C(=O)NCC(CCOC)NC(C2(CCOC)CCC2)=O)cc(C(F)F)ccn1 N1(C(CCc2onc(CC)n2)=O)CC2CC(C)N(C(=O)C(CO)C(C)(C)C)C2C1 O=C(C1=NOC2(CCC2)C1)NC1CC2(C1)CC2NC(C1CCC(F)(F)C1)=O c1(OCCC)cc(C(C)NC(c2cccc(C)n2)CC)ccc1OCCC c1(C(N2CC(CNC(CC(CC)C)=O)C(C)C2)=O)ccc(F)c(Cl)n1 Cn1nnnc1N1CCC(NCC2CN(S(=O)(=O)C(F)F)C2)C1 N1(CC(=O)N(CCOCCCNC(C2C(=C)C2)=O)C)CCNC(=O)C1 c1(CC(N2C(C(=O)NC(C(C)(C)OC)C)C3CC3C2)=O)ccc2c(c1)CC2 c1(N(C(c2ccccc2Br)C(F)F)C(=O)NC2CC(CBr)C2)ccc(F)c(Cl)c1 N1(C(c2cc(C)oc2)=O)CCC(C)C(CNC(=O)COC2COC2)C1 CCC(C)CC(C)C(=O)NC1CC(NC(c2ccccc2NC(=O)CC#N)=O)C1 CS(=O)(=O)c1ccc(C(N2CCOC3(C2)CN(C(c2cc(Cl)cs2)=O)C3)=O)cc1 C1(CC)C(CC(=O)NC(CNC(c2cc(C(=O)OC)on2)=O)C(C)C)C1(F)F c1(C(CCCn2cccn2)C2CC2)nnnn1C(C)C.C(C=O)OCCOCC O=C(C(O)CC1CCOCC1)NCC1(F)CC(NC(C23COCC2C3)=O)C1 c1(C(=O)NC2C(OC)CN(C(=O)CCC=C(C)C)C2)cc2ccc(F)c(F)c2o1 C1(C(=O)NCC2CCN(C(=O)CSCc3ncc[nH]3)C2)CCOC1C(F)(F)F c1(NC(C(C)C)CCN(C)C(c2cc3n(n2)CCC3)=O)cc(S(C)(=O)=O)ncn1 N1(C(CN(C(=O)Cc2cnoc2)CC#C)=O)CC2CCOC2C1 c1(C(=O)NC2CCCC(NC(COCCCOC)=O)C2)c2c(nn1C)CCSC2 c1(-c2n[nH]c3c2CN(c2c(C(=O)OCC)cccn2)C3)ccc2cccnc2c1 c1(NC)cccc(C(=O)N(CC(C)NC(c2ccnc(C(C)(C)C)c2)=O)C)n1 c1(C(=O)NCCC2(O)CN(C(c3nc(OCC)sn3)=O)C2)cnc(C)nc1C C1(CNC(CC=C=C)=O)CCC(C)N(C(c2ccc(NCCO)cc2)=O)C1 CCC(C)C(O)C(=O)NCC1CC(F)(F)CN1C(c1cc2occc2[nH]1)=O c1(C(N(C2CCCN(C(COCCCC)=O)C2)CC)=O)ccc2occc2n1 C1(N(C(C2CC(n3cc(C4CC4)nn3)C2)=O)CCO)CCC(CN2CCOCC2)C1 C1(OC)CCCCC1C(=O)NC(CNC(C1CC1(F)F)=O)C(C)C CC(C)(C(=O)NCC1(CNC(c2cn3ccsc3n2)=O)CC1)C(F)F C1(NC(N(CC)CC2CCC2)=O)SCCN1C(=O)OC(C)(C)C Cc1ncnc(C(=O)NCC2(C(=O)NCCC(C)(C)C)CCC2)c1C c1(C(=O)NC2CC(CNC(COCCOC)=O)C2)ccc(OC)c2c1CCCC2 C(=O)(CC(C)(C)C(F)F)N1CC(NC(=O)CCC(C)SC)CC(OC)C1 N1(C(=O)OC)CC2C=CC1C(C(=O)N(C(=O)CN1CCC13CCC3)C1CC1)C2 C1(CNC(C(CCO)N(C)C)=O)CN(C(C2CC(O)(C(F)F)C2)=O)CCC1(C)C n1(C(C)C)nc(C(=O)NCCn2cc(CN3C(C)CCC3C)nn2)cc1C(=O)O C1(NC(c2cccc(C(C)C)n2)=O)CC2CCC1N2C(=O)COCC1CC1 C(=O)(C1=CCN(C(c2c(C)nsc2C)=O)CC1)NCCC(CC)(F)F C1(C(N2C(CCNC(c3c(C)cc(C)o3)=O)CSCC2)=O)CC2C=CC1CC2 c12oc3c(cccc3c1C)NCC(C1CCC1)NC2=O.C1C(=O)N1.CCCOC c1(C(N(C)CCc2ccccn2)=O)ncc(C(F)F)cn1 Cc1nc(C)c(C(=O)NC2CCCC(NC(c3c(C)nsc3N)=O)C2)s1 N1(C(C2N(C=O)CCC2)=O)CC(C2CC2)(C(=O)NC2C(O)CC2O)C1 C1(n2cc(C3(OCC)CC3)nn2)C=CCC(C(=O)NC2CC(OCC)CC2O)C1 C1(C(=O)NC(c2cn(C)nn2)C)CCN(C(=O)CC2CCOCC2)C1C c1(C(N2CC3(CCC3)C2C2CC2)=O)ccc2c(c1)COCC2 C1(NC(c2coc(C(F)F)c2)=O)CCN(C(c2cc(O)nc(O)c2)=O)CC1CO N1(C(C(COC)C)=O)CC(NC(=O)C(O)Cc2ccccc2)CC12CCOCC2 Cc1[nH]nc(C(F)(F)F)c1C(=O)NC1C2CC1N(C(C1CCS(=O)(=O)C1)=O)C2 C1(C(N2CCCC(CNC(c3ccn(C)c(=O)c3)=O)C2)=O)CCOCC12CCC2 N1CCCC(O)(CO)C1.c1(OC)ccccc1NC1CC(CC(=O)NCCO)C1 c1(C(N(C2C(O)CCN(C(C(C)NC(N)=O)=O)C2)C)=O)ccc2cnsc2c1 c1(OC)ccc(F)c(C(=O)NC2(CCC(N3CCN(SC)CC3)=O)CCC2)c1F C(=O)(CC1=CCN(C)CC1)NCCN(C(=O)Cc1c(O)ncnc1O)CCOC c1(OCC)cc(C(N2CC(NC(C3COCCN3C)=O)CCC2C)=O)cc(F)c1 c1(C(=O)NC(C)CCCNC(=O)CC2CCCOCC2)cnc2n1CCC2 C1(NC(c2c(N=[N+]=[N-])cccc2)=O)CCCCC12CCN(C(C13CC1C3)=O)C2 CC1CN(C(C2C=CCC2)=O)CCCN1C(c1ccnn(C)c1=O)=O C1(CNC(CC(COC)C)=O)CN(C(C2CN(C)CCO2)=O)CCN1C Cc1cc(C(=O)NC(C)CCCCNC(c2cc(N)cc(O)n2)=O)c(Cl)cc1F c1(CNc2ccc(NC(c3cc(C)c(I)cc3)=O)c(F)c2)cccc(C#N)c1F C1(CC(=O)N(CCNC(C(C)(C)NC(C)=O)=O)CCNC(C)=O)CCCN(C)C1 c1(C(C)(C)OC)nc(CC(C)C)nn1-c1ccc(NC(N2CC(CF)C2)=O)cc1 C1(NC(c2cccc(CNC(c3n(C(C)C)ncc3)=O)n2)=O)CC2(CCCO2)C1 C=CCC(CC(C)C)C(=O)N1CCCC(CNC(c2cc(C)c(C)c(F)c2)=O)C1 c1(CC)ccc(F)cc1C(=O)NCC(C)CNC(=O)C=Cc1ccc(C(N)=O)o1 c1(C(C)C)ccc(Cl)c(NC(C2CN(C(c3cncc(Br)c3)=O)CC2C)=O)c1 c1(SC)cc(C(N2CCC(COC)(NC(=O)C=C3CC3)CC2)=O)c(Cl)cc1Cl N1(C(C2COCCN2C(c2cc(Cl)ncn2)=O)=O)CC2(CNC(=O)N2)C1 C(C(C)(C)CNC(c1ncsc1C)=O)C1CN(C(COCCCCC)=O)C1 N1(C(C(C2CCOC2)OCC)=O)CCC2(CCN(C(c3cn(C)cn3)=O)CC2)C1 O=C(C1=CCCCO1)NCCCN1CCN(C(C2C=CCS2)=O)CC1 C(=O)(C1=NOC2(CCC2)C1)NCC1CCC(N(C(=O)C(C)(Cl)Cl)C)CC1 Cc1nc(NCCC2(C)CCC2)cc(=NC(C)c2cc(O)n[nH]2)[nH]1 Cc1ccc(C(=O)NCC(N2CC(NC(=O)C(F)C(C)C)C2)=O)cc1 N1(C(C(CC(=O)OC)C)=O)CC2(CCC(CNC(c3ncc(N(C)C)cn3)=O)O2)C1 C1(C(N(CC(O)CF)CC)=O)OCCC1CNC(N)=O.C1(=O)CCCN1 N1(C(C(C)SC(C)C)=O)CC(C2CC2)(C(=O)NCCC2(C)CCC2)C1 c1(-c2n(CC(CC)CC)nc(Cc3cc(Cl)cc(Cl)c3)n2)cccc(Cl)c1OC n1(CC(=O)NC2CC2NC(C2CC23CC3)=O)ncn2cccc2c1=O C1(CC)CN(C(=O)C(O)CC(C)C)CCN1C(=O)C=CC1(C)CCOCC1 C1(C(=O)NC)CCN(C(C2(OC)CCN(C(=O)C(C3CCCCC3)C)C2)=O)C1C CC1CC(CS(=O)(=O)NCCCCC(=O)NC2CC2)CCO1 C(=O)(C(F)C(C)(C)O)N1C(C)(CC(=O)NCC2CCN(C)CC2)CC1 C1(NC(c2c(C)sc(Cl)n2)=O)CC2CC1N(C(=O)CCC(=O)c1cccnc1)C2 c1(-c2cn(CCC(N)=O)nn2)cccc(NC(=O)Cc2cccs2)c1 N1(C(CCC(C)OC)=O)CC(CNC(c2cc([N+](=O)[O-])n[nH]2)=O)C(C)(C)C1 Cc1nc(C(N2CCCN(C(c3cc(C#N)c[nH]3)=O)CCC2)=O)c2n1CCCC2 C(=O)(C(O)C(F)(F)F)NC1CC(C)(NC(c2c(C)nc(O)s2)=O)C1 c1(CNC(c2c(C(=O)OCC)cnn2C)=O)ccc2c(ccn2C)c1 N1(C(C(C)OC)=O)CCOC2(CCCN(C(=O)CC3(NC(=O)SC)CCCC3)C2)C1 c1(C(N)=O)cc(C(=O)NC2CCC(NC(C3CCCC3CF)=O)C2)on1 c1(C(=O)NCC(CNC(COCCCC)=O)(C)O)c(C)ccnc1C N1(C(C2CC=C(C)CC2)=O)CCCC(F)(CNC(=O)Cc2ccc(CO)cc2)C1 c1(OC)ccc(Cl)c(C(=O)N(CC(C)NC(=O)Cc2cnc(C)o2)C)c1N C1(C(N2C(COC)C(C)CC2)=O)C2CCN(C(C3CC(=O)CCO3)=O)CC12 CCCCC(C)C(=O)NCC(O)CNC(C1CSC1)=O Cc1cc(N)cc(C(=O)NC2COCCC2CCc2ccccc2)c1F Cc1csc(C)c1C(N1CC(C(=O)NC(c2cccc(O)c2)C)C(C)C1)=O C#Cc1ccc(C(=O)N(CC(C)NC(c2cc(C)ccc2F)=O)CC)c(OC)c1 c1(C(=O)NC(C)CN(C(=O)CC(C)(O)c2ccccc2)C)ccccc1C(C)O C=CCC(CNC(=O)C(C)CC1CC1)C(=O)NCCNS(N)(=O)=O n1(CC=C)nc(-c2ccoc2C)nc1-c1ccccc1Cl C12(CNC(CSC(C)C)=O)CCCC1N(C(=O)C(C(C)(C)C)SC)CC2 C1(C(=O)NCc2c(OC)nsc2)CCN(C(c2nscc2C)=O)C12CCC2 C(C1=CCCSC1)(c1ccc(Cl)cc1)NC(C(=O)NCC=CCSC)=O c1(C(=O)OC)cc(NC(=O)NC(=O)NCC(c2cnccc2C)(C)C)cc(Br)c1 Cc1[nH]nc2c1CC(N=c1[nH]c(NC3C4CCCC34)nc3c1CCCCC3)CC2 Cc1ccc(C(N2CC=CC2CNC(C2(Cl)CC23CCC3)=O)=O)nc1 c1(C(N(CC(C)(C)NC(=O)CCc2nccs2)C)=O)cc(O)cc(N)c1Cl C1(C)(C(=O)NCC2CCN(C(c3c(C)cnnc3)=O)C2)COc2ccccc2O1 C1(NC(c2ccc(SC)s2)=O)CC12CCN(C(c1ccc(CO)nc1)=O)C2 c1(OC)ccc(C)c2[nH]c(C(=O)NC3CC(N(C)C(C4CCOC4=O)=O)C3)cc12 N1(C(C(=Cc2cnc[nH]2)C)=O)CC(NC(=O)Cc2cnn(C)c2C)C(C)C1 CCCCC(CC)C(=O)N1CCC(C2CC2)C1CNC(c1ncc[nH]c1=O)=O C1(N(C(=O)C=CC2CCCO2)C)CCN(C(=O)Cc2nccn2C)CC12CC2 C(=O)(C(CC(C)(C)C)OC)N1CC(C)(OCC(=O)NC2CC(O)(CC#C)C2)C1 CCCCCCC(F)C(=O)N1CCC(CN(C(=O)C(O)CCC(C)C)C)CC1 c1(C(N2CC(CCCNC(C(C)SC)=O)OCC2)=O)cccc2nsnc12 Cc1nc(CNC2CC2)oc1C(N1CC=CC1CNC(=O)Cn1ccnn1)=O Cc1nc(C(F)(F)F)sc1C(N1CC(O)(C(C)NC(=O)C=C(Cl)Cl)C1)=O C(C)(C)(CCC(=O)NC1CN(C(=O)C(C)(C)COCC(F)F)C1)OC c1(OCC(=O)NC2C3CCN(C(c4nc(C)[nH]n4)=O)C32)ccc(S(N)(=O)=O)cc1 c1(OC)ccc(CCC(=O)N(CCN(C)C(c2[nH]nnc2C)=O)C(C)C)cc1F C1(C(N(CCCNC(c2cnn(C(F)F)c2)=O)CC)=O)CC2(CSC2)C1 C(=O)(C1CCCc2sccc21)N(CCNC(c1ccc(C)s1)=O)CC N1(C(C(C)Oc2cccc(Cl)c2)=O)CC2(C1)CN(C(=O)Cc1csc(=N)[nH]1)C2 C1(CC)CC(C(N2CCC(C(C)NC(=O)Cc3ccccc3)CC2)=O)CC(=O)N1 c1(C(=O)NC(c2ncc[nH]2)C)ccc(S(c2nnnn2C2(C)CC2)(C2CC2)CC)cc1 C12(NC(=O)C3=CCCCC3)CCCC1N(C(C13CCCC1(C(N)=O)C3)=O)CC2 c1(NC(N2CC(CO)OC3(CCC3)C2)=O)ccc2ccc(O)nc2n1 C(CCCCC(=O)NC1CCN(C(C2(CF)CC3(CCC3)C2)=O)CC1C)OC N1(C(C2OCCN(C(c3ccc(C)s3)=O)CC2)=O)CC(C2CCCCC2)C1 N1(C(C(C)C#N)=O)CCC(C)(C)C1CC(=O)NC1(C)CN2CCC1C2 C1(C(N2CCC(C(C(=O)Nc3c(C(C)C)n[nH]c3)C)C2)=O)CC(=O)NC1(C)C N1(C(c2c(CNC(CC3N(C)CCC3)=O)nnn2C)=O)CCC12CCC(O)CC2 C=C(Cl)CCC(=O)NC1CCCC1NC(c1ccc(N2CCC(O)C2)cc1)=O C1(NC(CC(C)NC(c2cnc(C3CC3)o2)=O)=O)CC(=O)N(C2CC2)C1 c1(OC)cc(C(=O)NCCCNC(=O)C(O)CC2CC2)cc(OC)c1OC(F)F c1(CO)ccccc1C(C(=O)O)N.n1(C(C)C(=O)N(C)C)cc(CCC2CC2)nn1 N1(C(CNC(N)=O)=O)CC(NC2CCN(C3CC3)C2=O)C2(CCC2)C1 Cc1ccc(C)c2[nH]c(C(=O)NC3CN(C(=O)CCCC(C)(F)F)CC3O)cc12 N1(CC)CCSCC1c1ccccc1.C1(F)(C(=O)O)CC1C(=O)NC1CCCC1 C1(CC)CN(C(=O)CCc2csc(C)n2)CCN1C(C)=O c1(C(N2CC(COC)(CNC(c3c(C)coc3C)=O)C2)=O)c(F)cccc1Cl C(C1CCC(C)CC1)=C(C)C(=O)N(C)CC1CC(F)CN1C(c1cc[nH]n1)=O C1(NC(c2ncn(CC)n2)=O)CC2CC1N(C(c1ncoc1C1CCCO1)=O)C2 CON(CCC(=O)N1CCC(C)(C)C1)C(=O)C1C2CCC(=O)C12 C1(CN(C(C(=O)NCC=C)C2CCSC2)C)CCCCO1 N1(C(=O)Cn2ccc(C(F)F)n2)CCOC(CNC(C2CC2(F)F)=O)C1 N1(C(c2cccc(CC#N)c2)=O)CC(NC(=O)COC(F)F)CC12CCCC2 C1(C(=O)NCCC(C)NC(c2cnn(CC)c2C2CC2)=O)CC2CC1CC2O C(=O)(C1=CCN(C(C2COC(C)C2)=O)C1)NCC(C)(C)SC C1(C(=O)NC(CN(C(C(c2cccc(Cl)c2)CC)=O)C)(C)C)CC2COCC2C1 C1(c2nc(-c3cccc(SCN4CCC(C)CC4)c3)on2)OC(C)(C)C(C)(C)O1 c1(C(=O)NCC2(NC(C(C(C)OC)O)=O)CCC2)ccccc1[N+](=O)[O-] N1(C(c2c(C(C)=O)coc2)=O)CCC(O)C(NC(=O)CCn2ccnc2C)C1 c1(C(C(=O)NCC(CNC(C2(OC)CCSC2)=O)OC)SC)ccccc1 N1(C(C2CCC(CNC(C(C)N(C(C)=O)C)=O)C2)=O)CCN2CCOCC2C1 C(CC(C)CC)(C(=O)N(C)CC12CCC(CC1)C2)NC(C1OCCN(CC)C1)=O C(CCC(C)NC(c1n[nH]c(C2CCCC2)n1)=O)NC(CCNC(COC)=O)=O C(=O)(CC(C)CC(F)(F)F)NC1CC(CNC(C(CC#C)C2CC2)=O)C1(C)C c1(C(N(CCCNC(C2(C)CC(F)C2)=O)C2CC2)=O)cncc2c(F)cccc12 Cc1[nH]c(=NCC=CCNC(c2occ3c2CCC3)=O)ccc1C#N N1(C(c2cc(C)nn2C)=O)CCOCC(C(=O)NCC(F)(F)F)C1 c1(C(N(CCNC(=O)CCC2CCCC2)CC)=O)ccc2c(c1)n(C)c(=O)n2C C1(OC)CC2(C1)CC2NC(=O)C(=O)NCCCC1CCCC1.c1(C)cccc(SC)c1 C1(CNC(c2ccc(-n3cnnc3)cc2)=O)CN(C(=O)Cn2ccnn2)C2CC12 C1(C(=O)NC(C(C)(C)NC(CC(C=C)(C)C)=O)C)CC2(CC(C)=NO2)C1 N1(C(C(C)CC(N)=O)=O)CCC(C(=O)NC(c2cc[nH]n2)C)=C(F)C1 CCCCCCCCCOC(Cc1ccc(C(O)CC)cc1)=O N1(C(C(C)C2CC2)=O)CCCC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])C1 C(=O)(CCC(C)NC(=O)C(C)(C)Cl)NC(CSC)C CON(C)CCCN=c1[nH]ccc(=NC(C)c2cc(C)oc2C)[nH]1 c1(C(N(CC(CNC(CCN(CCC)C)=O)C)C)=O)ccc(F)c2c1CCC2 c1(C(N(CCCNC(=O)Cn2cnnc2)C)=O)cc(NC(N)=O)ccc1Cl c1(C(C(=O)NC2C(NC(CCCCCCC)=O)CC2)C)cn(C)c2ccccc12 N1(C(C2(OC)CC2)=O)CCC(C2CCCN(C(=O)C3=C(Cl)CCOC3)C2)C1 C(=O)(CCC(=O)NCCCCCC)NCCC1(NC(CC=CC)=O)CCC1 c1(CC)ncoc1CNC(=O)C(C)(C)C1CCCN1C(c1ccn(CCF)n1)=O CC(F)(F)CC(=O)N1CCCC1CCC1CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 c1(C(=O)NC2(C(N(C)CC3CCCCCC3)=O)CC2(C)C)ccn2nccc2c1 C(=O)(C(C(C)C)NC(C1CC(CCNC(=O)C=Cc2ccsc2)C1)=O)NC C1(NC(Cc2nc(C)sc2)=O)CS(=O)(=O)CC1N=c1[nH]nc(C)o1 c1(C(=O)NC(CNC(c2cc(C(CC)C)no2)=O)(C)CC)ccc(C)cc1SC N1(C(c2cc(OCC)no2)=O)CCN(C(c2cc(C)cc(F)c2)=O)C(C)C1C N(C1COc2cc(Cl)ccc21)C(c1ccc(C=CC(F)(F)F)cc1)=O N1(C(CCc2cc(C)[nH]n2)=O)CCC(NC(C2CCC(=O)CC2)=O)C(C)(C)C1 C1(OC)(CNC(N2CCC(c3ccco3)C2)=O)CCNC1=O c1(OC)cc(C)c(C(=O)N(CCCNC(C2(F)CCOC2C)=O)C2CC2)cn1 N1(CCN(C(=O)Cn2cccn2)C)CCN(C(=O)CNC(N)=O)CC1 C12(CN(CCC)C(c3cccc(C(=O)OC)n3)=O)CC3CC1(CO)CC3C2 C(=O)(C1CCOc2ccc(F)cc21)N1C(CNC(c2c(C)nco2)=O)CCC1 N1(CC)C(=O)CCC1C(=O)NCC1(O)CC(NC(=O)CC2CCC2)C1 CCC#CCCNC(C1C(C)CN1C(=O)CC1CCCSC1)=O Cc1cc(C)c(S(=O)(=O)NC2CCC(NC(C3CCCN(C)C3)=O)CC2)c(C)c1 CCCCC(O)C(C)C(=O)N1CCN(C(c2cccc(C)n2)=O)CC1C CCC(C)CC(=O)C(=O)N1Cc2[nH]nc(C(=O)NCC34CCN(CC3)C4)c2C1 Cc1cc(OCCC(N2CCSC2CO)=O)ccc1Br C(=O)(C(C)(C)CS(N)(=O)=O)N1C(C)CC1CNC(=O)C(c1cccc(Cl)c1)O N1(C(=O)NOC(C2(C)N(C(=O)C3CC3)CCC2)=O)CC(CC)CCC1=O.O.O C1(C(N2C(C)(C(=O)NC)CCC2)=O)CCC(C)(C)N(C(=O)C(C)CC(F)(F)F)C1 c1(CC(=O)NCC(C)NC(=O)CSc2nc[nH]n2)cccnc1C(F)(F)F c1(C(=O)NC2CCCCN(C(c3ccc(C#C)cn3)=O)C2)ccc(C)c(C#N)c1 C1(NC(CCCSC)=O)CCC2CN(C(=O)C(=O)Nc3ncc[nH]3)CCC2C1 c1(C(=O)NCC(C)NC(=O)CCc2cncn2C)cncc2cnccc12 C(=O)(C(C)C(O)CCCC)NCC1(NC(C(CC#C)CC#C)=O)CCCCCC1 CC1CCN(C(c2ns[nH]c2=O)=O)CC1CNC(C1(CO)CCCCC1)=O CC(C(=O)N1CC(N(C)C(c2cnc(O)n2C)=O)C2(CC2)C1)C(C)(C)C C1(CNC(c2cccc(CO)n2)=O)CCCCC1NC(C12COC(CF)(C1)C2)=O N1(C(C(CC(C)C)C)=O)CC(C)(C)OC2(C1)CN(C(c1cc3sccc3s1)=O)C2 CC12CCC1CN(C(=O)C(c1cccnc1)NC(=O)C(c1ccccc1)F)C2 c1(C(=O)NC(CC=CC(=O)NC(c2ccnn2C)CC)(C)C)n[nH]c(CC)c1C C1(C(=O)NC(=O)Cc2ccco2)CCCN(C(=O)CCOCC(F)F)CC1F C1(O)(CC(=O)NC(C)C(CO)NC(=O)CCC2CCCCO2)CCCCCC1 c1(C(N(C)Cc2ccc(CNC(c3scc(C)c3)=O)cc2)=O)cncc(N)c1C c12ccccc1S(=O)(=O)N(CC)CCC(=O)N2.C(C)(C)(C)NN(C)C C=CC(C)(CC)C(=O)NCC1CCC1C(N1CCOC(C2CCC2)C1)=O c1(C(N(C)CC2CCN(C(=O)CC(O)c3ccccc3)C2)=O)cnc(Cl)c(N)c1 C1(C(=O)NCC)CN(C(=O)CCCOC)CC12CC2.C#CC12CN(C1)C2=O C(N=c1[nH]c(C#N)c(Cl)s1)C1CN(C(c2cn(CC(CC)O)nn2)=O)CC1C c1(-c2n(-c3ccn(CC)n3)nc(COc3ccccc3)n2)cccc(S(C)=O)c1 C1(NC(CNC(CCC)=O)=O)CC(C)N(C(c2n[nH]c(C)c2Br)=O)C1 C1(NC(CCSCC)=O)CCCN(C(c2cc(OC)cc(Br)c2)=O)C1C c1(C(=O)NC2C(OC)CN(C(=O)CSC)C2)ccc(C)c2cccnc12 c1(CC(=O)N(CCN2CCN(C(CC(CC)O)=O)CC2)C)cc(O)nc(O)n1 C1(Cn2ncc(C)c2)CCCN(C(C2CC3CCC2O3)=O)C1 c1(NC(C2C(O)CCN(c3nc(C)cc(SC)n3)C2)=O)nc(Cl)ccc1C#N C=C=CCCC(=O)N1CC(OCC(=O)NCCSc2ccc(F)cc2)C1 C1(C)(CNC(c2cnc(CCC)s2)=O)CN(C(C2CC(C)(O)C2)=O)CC1C c1(NCc2n(CC)cnn2)ccc(C(=O)NCCC2NC(=O)NC2=O)nc1 c1(C(N2CCC(N(C(C(=O)NCC#C)=O)C)CC2)=O)c(F)ccc2ccoc12 C1(OC)(CNC(=O)NCC2CCC(=O)NC2)CCC(C)(CO)CC1 Cc1nc(C(=O)N(C(C)CNC(=O)C(c2cccc(Br)c2)(C)C)C)c(C)o1 c1(NC)ccc(C(=O)NC2CCCC2CNC(=O)CC2(O)CCC2)c(Cl)c1 Cc1ncc(Cl)cc1C(=O)NC1CS(=O)(=O)CC1NC(C1CCCC(F)(F)C1)=O CCC(C)(CC(=O)NC(c1ccc(F)cc1F)CNC(=O)C=C(C)C)C(=O)OC N1(C(C(C)OCCN(C)C)=O)CC(C2CCCN(C(C3(C)CCC(=O)N3)=O)C2)C1 C1(C(=O)OC)CN(Cc2nc(C)cn2C)CC12CC2 N1(C(C(C(=O)OCC)F)=O)CC(CNC(c2cnc(C(F)F)s2)=O)CC1(C)C c1(CC(=O)NCC2CCCO2)ccccc1C(F)(F)F.c1(C(C)(C)C)cn(CC)nn1 C1(CN(C(c2c(CC)c[nH]n2)=O)C)CN(C(=O)C=CC2CCCO2)CCO1 c1(C(F)F)n[nH]c(=NC2CC3OCCC23)o1 C(=O)(CCC(F)F)NCCC(C)N(C)C(c1cc(Br)n(C)c1)=O c1(CN(c2ccccc2)C)cccc2c1CNCCC2.C1CCO1 C1(CNC(=O)NCC(CC)(C)c2ccccn2)CN(C)CCN(C)C1 C(C(CNC(=O)CC1(N(C)C)CC1)S(C)(=O)=O)NC(C(CC)OCC)=O c1(OC)ccc2cc(C(=O)NC(CNC(C3C4CCCC34)=O)CC(C)C)sc2c1 Cc1ncc(C(=O)NCC2(O)CCCN(C(c3nnsc3N)=O)C2)cc1Cl Cc1noc(C)c1CN(C(=O)C(Cn1cccn1)NC(=O)C(C)OCC1CC1)C Cc1ccc(CC(=O)NCCC(C)NC(=O)C(F)(F)c2cnn(C)c2)cc1 C(C(C)CNC(C1(CCN(C)C)CC1)=O)NC(C1C(=C)C1)=O Cc1csc(=NCC(=O)N2CCC3CC3(NC(=O)CCn3cccn3)CC2)[nH]1 c1(C(=O)NC2(CNC(C3(C)CC(C)C3)=O)CCOC2)cc(C(C)(C)C)nn1C C(=O)(C(C)CC(=O)c1ccccc1F)NCC1(O)CN(C(c2c(C)nsc2)=O)C1 N1(C(C(CSC)C)=O)CCC2OCCN(C(c3cc4cccnn4n3)=O)C2C1 C1(CNC(=O)C=C(Cl)Cl)CC2COCC2N1C(=O)CN1C(=O)CNC1=O C(=O)(C1=CC2C=CC1C2)N(C1CCN(C(=O)CCOC2CCC2)C1)CCOC(C)=O CN1CC(NC(c2cn(CCF)nn2)=O)C(C(=O)O)C1 c1(C(=O)NC2CC(F)(CNC(C3C(N(C)C)CCC3)=O)C2)ccc2scnc2c1 c1(SC)cccc(C(=O)NCC2CCCCN2C(c2cccnc2O)=O)c1Cl C1(NC(C(CC)C(C)C)=O)CN(C(=O)CCc2cn[nH]c2)CC2(CCC2)C1 N1(C(COCC(=C)C)=O)CCCCC1CCNC(c1csc(C)n1)=O c1(C(=O)NCC(C)(C2CC2)NC(c2ccsc2)=O)ccc(Cl)c(F)c1 C1(C(NOCC#C)=O)CCC(C)(C)N(C(=O)COCCN(C)C)C1 CC(CCC(=O)NCCC1CCC(C)(C)O1)NC(c1ccon1)=O c1(C(=O)NC(C)CNC(c2cc(N)cc(O)c2F)=O)cc2c(F)ccc(F)c2[nH]1 C1(NC(C(c2cccc(O)c2)C)=O)CC12CCN(C(=O)C(C)(C)N(C)C)CC2 c1(CC(N2CCC(N(C(=O)C3=CCSC3)C)CC2)=O)coc2c(F)c(F)ccc12 c1(NC(C2CCN(C(=O)OC)C2)=O)ccc(OC)nc1.c1(COCC)ccccc1NC c1(CC)c(OC)cccc1C(N1CCN(C(=O)CCCn2cncn2)CC1)=O c1(OC)cccc(N2CCC(NC(=O)CSc3nc(C)c(Br)s3)C2)c1 c1(N(C(CCN(C)CC=CC(=O)NC(C)C)C)C)nc(C)ncc1Cl C1(NCc2c(CNC(C3(C)CC3C(F)(F)F)=O)cccc2)CCC=CCCC1 c1(C(=O)NC2CC(C)(NC(=O)CC3CC3)C2)cc(O)ccc1Br C#CC1(C(=O)NCC(C)C(=O)NCC2(O)CC2)CCCCC1 C1(C(C)(C)NC(c2c[nH]nc2C2CCCO2)=O)CCN(C(=O)Cc2ccon2)CC1 C#CC1(C(=O)NCC2CCC(C(=O)NC(C)C(O)C(F)F)C2)CCCC1 C(=O)(C1=CCCSC1)NC1CC(C(C)NC(CCCCOC)=O)C1 N1(C(C2(CC)CC2(F)F)=O)CCC(O)(CCNC(c2cncc(O)c2)=O)C1 C(CNC(=O)C(Cl)=CCl)(C(C)C(C)C)NC(c1c(CSCC)cccc1)=O C1(COC(c2c(CC(=O)OC(CC)(C)C)c[nH]n2)=O)CC(CO)N(C)C1 C1(NC(Cc2c(C)oc(-c3ccco3)n2)=O)CCCCN(C(=O)C(C)C#N)CC1 N(C1CCCn2nccc21)C(=O)CC1CN(C(=O)CSc2nc[nH]n2)CCO1 CC1CC(NC(C2CCC2NC(c2cc(O)ncc2F)=O)=O)CC(C)(C)C1 Cc1c(CS(=O)Cc2ccc(F)cc2)noc1C1CC1 N1(C(=O)NCc2cnc(CC)s2)CC2CCC(C(=O)OC)(C2)C1 Cc1cc(=NCC2CCC(F)(F)C2)[nH]cc1S(=O)(=O)NC1CCOCC1C(N)=O C(C(C)(C)C(C)(F)F)C(=O)NC1(C)CCN(C(c2c(OC)scc2)=O)C1 C1(CNC(C(=O)OCC)Cc2nccn2C)CC12CCOCC2 C(=O)(CCSC)NCCN(CCOC)C(C1CC1(Cl)Cl)=O C(=O)(C1=NOC(C)C1C)N1CCC(C(=O)N(c2ccccc2O)C)(OC)C1 C(=O)(C(C)(C)C(C)(C)O)NCC(C)(C1CC1)NC(C(CC1CCC1)OC)=O Cc1ccc(CC(=O)NCc2ccc(-c3ccccc3)nc2)cc1Cl N1(C(C(CCC)=CCC)=O)CC2(CC(NC(c3ccc(OC)o3)=O)CO2)C1 N1(CCN=C(NCC2(COC)COC2)NCC(F)F)CCCC(C)(C)CC1 NS(=O)(=O)c1ccc(CC(=O)NCC2CN(C(=O)CCCCCF)CCCO2)cc1 CN1CC=CCC1CC1CCN(C2CC3(C(=O)NC)CC2C3)CC1 O=C(C1=CCCOCC1)NCCCCCNC(C1CCC2(C1)CC2(F)F)=O C=C1CC(CC(=O)N(CCC)CCNC(C2CC2(C)CSC)=O)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N1C2CC(CNC(c3c(C)nc(C)n3O)=O)C1CC2 c1(CC)cc(N(C2CCN(C(=O)CCC(C)(F)F)CC2)CC2CC2)nc(C)n1 Cc1cc(Br)cnc1CNC(=O)Nc1ncc(F)c(=N)[nH]1 c1(C(c2n(C(CC)C)nnn2)NCc2ccncn2)cc2ccccc2s1 C1(NC(CCCCC#C)=O)CN(C(=O)C2=C(C#N)CCC2)CC12CCOCC2 CC1CCCC=C1C(=O)N1CC(NC(=O)CSc2ccc(C#N)cc2)C2(CC2)C1 N1(C(C2ON=C(C)C2C)=O)CCC2CCC(C1)N2C(=O)CCc1cccc(O)c1 N1(C(Cn2c(C)nc(C)n2)=O)C(C(=O)NCC(C)C2CCC2)CCC12CC2 C1(C(=O)NCC(C)CC2CCC2)(NC(COC)=O)CCC(C)(C)C1 c1(CC(C)(C)CO)nc(-c2cn(C3CCOC3)nn2)n(C2CCCSC2)n1 N1(C(=O)OC(C)(C)C)CCC(CNCC2CCC2c2ccccc2)C1 c1(C(N(C2CN(C(CCCC#C)=O)C2)C)=O)ccc(OC(F)F)cc1F CC(CN=c1[nH]c(N2CCOC3(CC3)C2)nc2c1SCC2)C(C)(F)F.CC Cn1nnnc1CCCNC(C1(NC(=O)CC2CC2C2CC2)CC(F)C1)=O C1(C(N(C)CC2CC2)=O)CC2(CC2)CN1C(c1c[nH]cc1C(C)(C)C)=O N1(C(C(CC=CC)C)=O)CC2(CNC(=O)C#CC3CC3)CCC1C2 N1(C(c2c(F)ccc(N)c2)=O)CCOC2CCN(C(=O)COCC(F)F)CC12 Cn1nc(C(F)F)c(CNC2CC(F)CN(C(c3cccc(Br)n3)=O)C2)c1Cl c1(OCC(=O)NC2CN(C(CCC3CCC(C)O3)=O)C2)cc(Cl)cc(Cl)c1 Cc1c(Cl)ccc(C(N2C3CN(Cc4cnc(C(=O)O)nc4)CC23)=O)c1F N1(C(CN(C(C(C)C)=O)C)=O)C2CCC1CN(C(C1CC1[N+](=O)[O-])=O)C2 C1(C(N(CCNC(=O)CCN2CCCCC2)C2CC2)=O)C(Cl)(Cl)C12CC2 C1(C(C)C)(NC(c2nnc(CO)s2)=O)CCN(C(=O)CN2CCN(C)CC2)CC1 c1(C(=O)NC(CCC)CNC(=O)CC2(NC(C)=O)CC2)cn(C)c(C)n1 c1(C(N2CCC(C)(NC(C(C)C)=O)CC2)=O)nccc2ccncc12 C1(NC(C2(Br)C(C)(C)C2)=O)COC2(CCN(C(c3ccncc3)=O)CC2)C1 c1(CCC(=O)N(C(C)CO)CCC)cc2ccc(O)cc2oc1=O C#Cc1ccc(C(=O)NCC(C)N(C(=O)C(c2cc(Br)co2)=O)C)cn1 N1(C(C(C)(C(C)C)OC)=O)CCC2(CCCN2C(c2csc(F)c2)=O)C1 c1(NC(C2(F)CN(C(Cc3cc(C)no3)=O)C2)=O)cc([N+](=O)[O-])ccc1C Cc1cc(C(N2CC(NC(=O)CCCc3cccs3)C(F)C2)=O)oc1C N1(C(C2N(CC)CCC2)=O)CCC(C2(NC(=O)CCc3cnn(C)c3C)CC2)C1 Cc1cc(N2CCC(CNC(c3cccn3Cc3cccs3)=O)CC2)nc(Cl)n1 c1(CC(C(=O)NCCC(CNC(CCN(C)CC)=O)O)(C)C)ccc(F)c(F)c1 C1(CC)CCOCCN1C(=O)CC1N(C(=O)Cn2cc(C#N)cn2)CCC1(C)C C1(CNC(=O)Nc2cccc(C(F)(F)F)c2)(NC2CCS(=O)(=O)C2)CCCCC1 C1(CC(=O)N(CCC(=O)NCCC2(C)CCCC2)CC)CCC(C)(C)C1 N1(C(c2nc(CC)oc2)=O)CC2CCC(C1)N2C(c1ccc(Cl)c(Cl)c1N)=O C(=O)(CC(O)CNC(=O)CC1CCC=CCC1)NC1(C)CCOC1 CC(C)(O)CC(CC(=O)NCC1CC1c1ccccc1)C(=O)O C=C1CCC(C(=O)NC2CN(C(=O)Cc3cc[nH]c3)CC2n2cccn2)CC1 CCC(C(=O)N(CCN(C(C1CC(n2cnnc2)C1)=O)CC)CC)C(C)C N1(C(COCC(=O)OC)=O)CCC(C)(C)C(NC(=O)CC2C=CCCC2)C1 N1(C(CN(C(C)=O)C)=O)CC(NC(=O)C2CC2)C2(CCS(=O)(=O)CC2)C1 c1(C(N2CCC(NC(c3c(CC)ncs3)=O)C(F)C2)=O)ccc(F)c(C#N)c1 CC1CCC(N=c2[nH]c3ccc(S(=O)(=O)NCCSCO)cc3s2)C1.C(F)(F)(C(F)(F)F)O c1(CN(C(=O)CN2CC=CCC2)C)ccc(F)c(F)c1 n1(CC)c(C)cc(C(=O)NC2CC2NC(c2cnc(C)nc2C)=O)c1C c1(C(N2CC(CC(=O)N(CC(C)C)CCC)C(C)C2)=O)nccc2[nH]ccc12 C1(C)(COC)CCN(C(c2cc(CNC(C3CCOCC3)=O)cs2)=O)CC1 c1(C(C2CCN(C(CCCn3cc(CC(C=C)O)nn3)=O)C2)C)ccccc1Cl N1(C(CN(C(COC)=O)C)=O)CC2CC2(CNC(C23CC(C)C2C3)=O)C1 c1(NC(C2CCN(C(C(C=CCCC)O)=O)CC2)C)cc(C)nc2c(C)cnn12 N1(C(C2CC23CCC3)C(=O)NCCC#N)Cc2cncnc2C1 c1(C(C(=O)NCCN(C(C2SCCS2)=O)CC)OC(C)(C)C)ccccc1 N1(C(C(CC=C)(C)C)=O)CCC2(C1)CN(C(c1ncc(Cl)n1C)=O)CCO2 c1(C(N2CCCC(C(C)(C)C(=O)NCC#CC#CCO)C2)=O)ccc(O)c(F)c1 c1(NC(c2c(NC(C)=O)cccc2)=O)cc(Cl)cc(C)c1[N+](=O)[O-] C(C(CO)CN=c1cc(C)[nH]c(-c2cnn(C)c2)n1)NC(C(C)OCCOC)=O c1(C(=O)NCCC(CNC(C(C2CC2)OC)=O)O)cc(C)n(C2CC2)n1 C1(N(c2ncncc2Cl)C(c2c(C)scc2)=O)CCCCC1c1nc(C2CC2)no1 CC(C)C1=NOC(C)(C(N2CCN(C(C3CCNC(=O)C3)=O)C(C3CC3)C2)=O)C1 C1(C(N(CCOCCN(C(C(CC)C#N)=O)C)C)=O)CCCC2(CC2)C1 C(C(C)CC(=O)N1CC2C(N(C)C(c3cnn(C)c3C)=O)C2C1)OC c1(CNC(c2ccc(CNC(CC=CC)=O)o2)=O)ccnc(O)c1 c1(C(=O)NCC23N(C(c4cc(C)[nH]n4)=O)CC(CC)(C2)C3)c(N)cc(Cl)cc1F n1(CCCC2N(Cc3n(C)cnc3I)CCC2)c(=O)oc2ccccc12 N1(C(C2CC(CC)OCC2)=O)CC2CCC(N(C(=O)Cn3cnnc3O)C)C2C1 c1(NC(C2C(NC(=O)COc3ccccc3)C2)=O)ccc2nn[nH]c2n1 Cc1ccncc1C(=O)NC1(C(=O)NCCC2CCCC3CC23)CC(O)C1 C(=O)(C1=Cc2cc(C)ccc2OC1)N1C(CNC(CSC)=O)C(C)(C)CCC1 c1(C(=O)NC(CN(C(C(c2cccs2)SC)=O)C)(C)C)cc2c(cn1)OCCC2 Cc1ccccc1-c1nc(CN(C)Cc2ccccc2)n(C2CCCCCC2)n1 C1(C(N2CC(F)(CNC(C3C(C#C)C3)=O)C2)=O)Cc2cc(C)ccc2S1(=O)=O N1(C(c2csc3nccn23)=O)CCCC(C2CN(C(C34CC(O)C3C4)=O)C2)C1 c1(CC)c(C(N2CCC(C)(NC(c3ccn(CC)n3)=O)C2)=O)cnn1CC(C)C c1(C(N(CCCCCNC(CSCCC)=O)C)=O)cc2c(cc1Cl)OCCO2 N1(C(C(CC)CC)=O)CCC2(CC1)CC(OCCn1cc(COC)nn1)CCO2 C1(NC(c2c(C)nc(C(C)C)o2)=O)Cc2cncn2C1 C(N=c1cc(NCC2(C(F)(F)F)CCC2)nc[nH]1)C1(C)CCC(F)(F)C1 N1(C(C)C(=O)O)CCN(C(=O)CC2CCCC(F)(F)C2)CC1=O N1(C(c2c(C)cco2)=O)CC2CCOCC2(NC(c2ccc(C(C)C)cc2)=O)C1 c1(C(=O)NC(CNC(C(C(CC)O)C)=O)CC)ccc2cnnc(O)c2c1 Cc1nc(C(C)NCc2ccc(OC(F)(F)F)o2)c(C)o1 c1(C(N(C2CCN(C(=O)CC(=O)N(C)C)C2)CCC)=O)oc(C2CC2)nc1C C1(C(N(CCn2cc(CC(O)C(C)C)nn2)CC)=O)CCC(C)(C)OC1 N1(C(CSCC(=O)OC)=O)CCCCC1CCNC(c1cccs1)=O Cc1cc(C#N)cnc1C(=O)NC1CC2(C1)CN(C(c1cnc(C(F)F)s1)=O)C2 Cc1noc(C2CC2)c1C(N1CCN(C(C2CCC(=O)N2C)=O)CC1)=O c1(C(=O)NC(CNC(c2ccon2)=O)C2CCC2)nnn(C2CC2)c1C(F)F c1(C(N)=O)csc(CCCNC(c2nnnn2C2COC2)c2ccccc2)n1 Cc1cc(F)ncc1C(N1CCC(O)C(NC(=O)Cc2cccc(Br)c2)C1)=O Cc1nccc(C(N2CC(N(C)C(C34CCN(CC3)C4)=O)C(C)(C)C2)=O)c1N N1(C(c2c(C)nc(CO)s2)=O)CCOCC(NC(C2CCC(CO)CC2)=O)C1 C(CCC[Si](C)(C)C)CN(C(c1ccc(CC2NC(=O)NC2=O)cc1)=O)CC C#Cc1ccccc1CC(N1CCCC(N(C(C2CC2F)=O)CC)C1)=O N1(C(C(C(=C)Cl)(C)C)=O)CCC2(CC1)CCN(C(c1cc(=O)n(C)cn1)=O)C2 C(CC(C)(C)C(=O)N1CCOC(C(=O)NOCC23CCC(CC2)C3)CC1)SC c1(C(C)(F)F)ccccc1C(=O)NCC1CCCCN1C(C1CC1C(F)F)=O C=C1CCN(C(c2cnn[nH]2)=O)C(C(N2CC(CC)CC(C)C2)=O)C1 Cc1c(C(=O)NCC2CCC(NC(=O)C=CC(N)=O)CC2)oc2ccccc12 C1(C(N(C)CC2CCOC2)=O)(NC(=O)NC2CN(C(N)=O)C2)CCN(C)C1 c1(C(=O)NC2CCCC(NC(c3cccc(C)c3F)=O)C2)cc2cccnc2[nH]1 CC(C)CC(O)CC(=O)N1CCOCC1CCNC(c1n[nH]c2c1CCCC2)=O c1(CNC(C23C(c4ccccc4)C2CC3)C)cc2n(n1)CCCC2 C(CCCCN=c1[nH]ccc(=NCCc2ccc(Cl)cc2OC)[nH]1)OC c1(NCCCCNC2CC(OC)C23CCC3)ccc([N+](=O)[O-])c(C#N)c1 C(=O)(C(C(=O)OCCCN(C)CCn1nc(C(F)F)cc1C)OC)OC c1(C(N2CCC(NC(C3(O)CCN(CCF)C3)=O)C2)=O)cc2ccccn2c1 N1(C(C(C)O)=O)CCN(C(c2n[nH]c(COc3ccc(F)cc3)n2)=O)CC1 CC1CC(NC(=O)Cn2ccnn2)CCN1C(=O)C(=O)C(C)(C)C CC1CC=C(C(=O)N2CC3(CC(C(=O)NC4(C5CCCCO5)CC4)CO3)C2)CC1 c12cncc(c1)C(=O)NC2.C1(CCC(=O)NC2CC(F)(CF)C2)(OC)CCCC1 C(=O)(CC(C)C(C)(C)C)NC(CCCC)CNC(=O)C(=Cc1cccs1)C c1(OC)cccc2c1OCC(C(=O)NCC(C(C)C)NC(C1(C)CSC1)=O)C2 c1(N2Cc3c(=N)[nH][nH]c3C2)nc2c(c(=NC3CCC4CC4CC3)[nH]1)CCCCCC2 CN1CC(C2CCN(C(c3cn(C4CN(c5cncs5)C4)nn3)=O)CC2)CC1=O CCC(CC)(CO)C(=O)NCC1C=CCN1C(=O)CCCn1cncn1 N1(C(C(CNC(=O)OC(C)(C)C)C(C)(C)C)=O)CCC2CN(C(=O)CCF)CCC12 C1(C(C)(C)C)(C(=O)NCC(CO)NC(=O)Cn2cnnc2O)CCCC1 C(C(C(C)C(C)C)NC(=O)C(=O)NCCC(N)=O)NC(c1c(CC)n(CC)nc1)=O C(C(C)(C)C(=O)NCCCCCN(C(=O)CC1CC2(CC2)CO1)C)N(C)C C1(NC(C(C)OC)=O)C2CC1N(C(c1cn(C(C)(C)C)nc1Br)=O)C2C C#Cc1ccc(C(=O)NCC2(C(=O)NC3CN(C4CCC4)C3)CCCC2)cc1C c1(C(N(C2CCCCN(C(C3CC3(F)F)=O)C2)C)=O)cc2ccncc2c(O)n1 CC1CCC(C(=O)NC2(CN(C)C(c3cnns3)=O)CC2)C(=O)N1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)N(CC(C)NC(c1ccc(Cl)c(Cl)c1)=O)C c1(C(N(C2CCN(C(=O)C=C3CC3)C2)CC)=O)ccc(OC(F)F)cc1F N1(C(c2c(C)ncnc2)=O)CC(CN(C(=O)C(C)(C)C2CCOC2)C)C2(CC2)C1 C1(CC(N2C(COC)C=CCC2)=O)C2CCCC2N1C(c1ccc([N+](=O)[O-])[nH]1)=O C(=O)(CC1=NNC(=O)C1)NCCC(C)(C)NC(C1(C)CCCC1(F)F)=O C12(O)CCN(C1)C2=O.C(C(=O)NC(C)(C)C)(c1cncs1)N(C)C N1(C(CC2OCCN(C(C=CC)=O)C2)=O)CC2CC(C)C2C1 N1(C(C2C3CC(OC)C(CC3)C2)=O)CCC2(CCC2NC(c2cccs2)=O)CC1 Cc1nc(C)c(C(N2CCOC(CN(C(=O)Cc3cnc[nH]3)C)C2)=O)[nH]1 C12(NC(CN(c3ccc(F)cc3)C(c3c(CC)occ3)=O)=O)CCC(C1)OC2C c1(C(C(=O)NC2CN(C(CCC=C=C)=O)C(C)C2)(C)C)ccc(F)c(F)c1 CC(CCC(=O)OC(C)(C)C)NCC1CCC2CC2C1 c1(NC(c2scc(C(=O)Nc3cncc(C)c3)n2)=O)ccc([N+](=O)[O-])cc1C N1(C(CC(CC)C2CC2)=O)CCC(C2(NC(C3CCOC3C)=O)CC2)CC1 c1(OC)cncc(C(N2CC(N(C)C(c3ccn(C)c3)=O)C2)=O)c1 C(=O)(NNc1c(Cl)cc(Br)cc1Cl)NCC(c1ccc(OC)c(OC)c1)O C1(C(N2CCC(CN(C(C(CC)=CCCC)=O)C)CC2)=O)CN(C)C(=O)CCO1 C1(CC(=O)NCC(C)CN(C)Cc2cc(C(=O)NC)no2)(CO)CCCCC1 C1(C)(CC)CCC(NC(=O)CNC(c2cccn(C)c2=O)=O)CC1 N1(C(C2(OC)CCC(C)(C)C2)=O)CCC2CCC(C1)N2C(c1csnn1)=O c1(OC)cc(Br)cc(F)c1C(=O)Nc1sc(-c2cnn(CCN(C)C)c2)nc1C C1(CNC(COCCCC#C)=O)C(C)CCCN1C(c1cc(=O)n(C)cn1)=O c1(C(C)NC2CCCCN(CC(=O)NC(C)(C)C)C2)ccc2ncsc2c1 c1(C(=O)NCC2COCCN2C(C2(F)CCC2)=O)cnc2ccc(Cl)cn12 C(=O)(CC(C)CC(=O)OCCC(C)C(F)(F)F)N(CC(=O)OC)CCOC C1(NC(C23C(C)(C)OCC2C3)=O)CC2CCC1CN(C(=O)Cc1c[nH]nc1O)C2 c1(CC)nc(C)oc1C(N1C(C(=O)N(c2cnn(C)c2C(N)=O)CC)CC2CC12)=O C1(C#N)(CN(C(CN(C(COCC(=C)C)=O)CC2CC2)=O)C)CCC1 c1(C(C(=O)NC(CC)CNC(c2c[nH]nc2C2CC2)=O)C)ccc(Cl)cc1 C(CNC(=O)C(c1cccc(Cl)c1)O)(CC(F)(F)F)NC(c1cc(C)c(C)[nH]1)=O C1(N(C(C2CCN(C(C3CCCN(CC)C3)=O)C2C)=O)CC)CCCC(F)(F)C1 C1(C(=O)NCC2C(C)CC2)(NC(=O)CC2CSCCO2)CC(F)(F)C1 c1(C(N2C(C)CCC(NC(C34CCN(CC3)C4)=O)C2)=O)ccc2nncn2c1 c1(C(CO)NC(C(=O)NCCc2cc(C(C)(C)C)no2)=O)ccc(Cl)cc1F c1(SC)cc(NC(c2ccc(F)c(C)c2F)=O)ccc1[N+](=O)[O-] N1(C(C=NOC)=O)CCC2(CCCN2C(C2C(COC)CC(O)C(O)C2)=O)C1 C(=O)(C(C)(O)c1ccccc1)N(C(C)CNC(=O)C(O)CC1CCOCC1)CC c1(C(N(CCCNC(=O)CC2C=CCCC2)CC)=O)cc2c(=O)[nH]ccn2c1 C1(C(N2CCCC(C=C)C2)=O)CN(C(c2c(C)ncnc2C)=O)CCC1(C)C Cc1cc(C(F)F)oc1C(=O)NC1CCC1NC(=O)C(C)(C)n1cnnn1 CC(CCCNC(C1CC1(F)F)=O)NC(c1cnc(-c2ccoc2)s1)=O C=C(C)CC(C)C(=O)NC1CCC(NC(c2ccc(OCC)cc2C(F)F)=O)C1 C1(CC(=O)N(C)CC2COCCN2C(=O)Cn2cccn2)CCC(C)(C)CO1 N1(C(Cc2cc(C)on2)=O)CCCC12CCCN(C(c1nocc1C1CC1)=O)C2 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CC=C(CNC(c2ccnnc2Cl)=O)CC1 Cn1cc([N+](=O)[O-])c(=NCC2CN(C(=O)CC3COC(=O)C3)CC2(C)C)[nH]1 CCC(C)C(c1nnnn1C(C)C)Nc1cnn(CC(C)C)c1 C(CO)(C(=O)N(C)Cc1cccnn1)NC(COCCC(C)C)=O c1(OC)cccc(NC(=O)C(C2(O)CCC2)NC(=O)CC(C)SC)c1 CC(C)CC(CC(C)C)C(=O)N1CCC(N(C)C(c2cc(Cl)ccc2O)=O)C1 c1(CC=CC(=O)NCCC(C)NC(C(C)C2CC2)=O)ccc(Cl)cc1 N1(C(CC2(C=C)CCC2)=O)CC(NC(=O)COC(F)(F)F)C(O)C1 c1(OC)ccnc(C(N2CCOC(CN(C)C(C3(C(N)=O)CCC3)=O)C2)=O)c1 C(C)(C(=O)NCC(C)(C)NCC(N1CC=CC1)=O)NC(=O)NC N1(CC(N2C(CNC(c3cc(COC)sc3)=O)C(C)CC2)=O)CCCCCCC1=O N1(C(CC2CC(OC(C)(C)C)C2)=O)CC(F)(F)CC1CNC(=O)C(C)CC(N)=O C#Cc1ccc(C(N2CCC(N(C)C(c3sc(C)nc3C)=O)CC2)=O)o1 CC(=O)C(C)CC(C)C(=O)N1CC(F)CC1CC(=O)Nc1ccccc1C1CC1 CCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(C1(F)CCC1)=O C1(NC(c2c(C(C)C)n[nH]c2)=O)C2CCC1N(C(=O)C(C)(C)c1cccnc1)C2 C1(NC(CS(=O)(=O)OCCOC)=O)(OCC)CCN(C(=O)C=CC(C)(C)C)CC1 C1(NC(=O)C(F)n2cccn2)CN(C(C2CC(n3ccnn3)C2)=O)CC1C(F)F N1(C(=O)CN2CCCCS2(=O)=O)CCC(C2CCN(CCCC3CCC3)CC2)C1 C1(OCC)CN(C(C2(C(F)F)CCCC2)=O)CC1CNC(C1CC2CC2C1)=O C1(CCNC(CC)=O)C(C)CCCN1C(=O)Cc1ccc(C(C)=O)cc1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(C1)CN(C(C1C=CCS1)=O)C2 c1(C(N(C)CC2CCN(C(c3cc(C(=O)OC)[nH]c3)=O)C2)=O)n[nH]c(CO)c1Cl c1(C(N2CCCC(NC(C3(CC#C)CCCO3)=O)C2)=O)cc(C(C)C)ccc1O C1(C(N(CC(=O)NCCC2CCCCO2)C)=O)CC2CC(=O)C1O2 c1(CN(C(C2(CCNC(c3cncnc3)=O)CC2)=O)CC)ncn(C)n1 c1(COCCNC(=O)NC(CC2CC2)C(=O)N2CCCC2)ccc2c(c1)CC2 N1(C(=O)NC2(C#N)CCCC2)CCN2CCOCC2C1 C1(CNC(CN2CCC(C)CC2)=O)CC2(CC2)CN1C(C12CC(F)(C1)C2)=O C=CCCCCC(=O)N1CCC(CC(=O)N(CC(O)COC)CC)C1 C1(CC(=O)NC(C=C)(C)CC)CC(C)(C)CN1C(c1sc(O)nc1C)=O c1(C(=O)NC(C)(C)CNC(=O)CSCC2CCCCO2)cccc2ccsc12 N1(CCc2cn(C3CCN(C(C4C(OCC)C4)=O)C3)nn2)CCCNS1(=O)=O c1(C(N2CCN(C(CC3CC(=C)C3)=O)CC2CC)=O)ccc(Cl)c(OC)c1F CC(C)CCC(F)C(=O)NC1CN(C(=O)C(=CC2CCCCC2)F)C2(CCC2)C1 CCC(C(=O)N1CCC(NC(=O)C(c2ccccc2)N(C)CC)C1C)C(C)C N1(C(Cc2c(OC)nccc2)=O)CC(NC(C2CC2C2CC2)=O)CC1(C)C C(C)(C(=O)NCc1cc(C(=O)NC2CCCCC2)n[nH]1)(C(C)C)OC C1(NC(C(C(C)C)NS(C)(=O)=O)=O)CCN(C(c2nocc2C2CC2)=O)C(C)C1 C1(C(=O)NC2CCC(CN(C(CCNC(=O)NC)=O)C)CC2)CCN(C)C(=O)C1 C1(n2cc(CCOC)nn2)CC2CCC(C1)N2C(=O)CC1CC(C(F)F)C1 CCC(C)(C(=O)NCCCOCCN(C(=O)C(CCOC)C1CC1)C)OC c1(C(=O)NCC(CCCC)NC(=O)C#CC(C)(C)O)c(C)nn2cc[nH]c(=O)c12 C=CCCN=C(NCc1cnn(CC)c1)N1CCCC(C)(C#N)C1 C(C1CCCC1)=C(C)C(=O)N(CC(O)CNC(C1CCCN1c1nccs1)=O)C n1(CCC(C)C)cc(C(=O)NC2C(NC(=O)CSc3cc(F)n[nH]3)COC2)nn1 Cc1c(C(=O)NCC2CN(C(C3CC(C)C3)=O)CC23CCC3)nn2c1CCCC2 c1(CN)ccc(-c2nn[nH]n2)c(C(F)(F)F)c1.N12CC(C(=O)O)C(C1)NCC2=O CC(CC(F)F)C(=O)OCc1nc(C(=O)NCCOc2ccccc2)co1 c1(C(=O)NC(C2CCCN(C(C3(CC(C)C)CC3)=O)C2)C)cn2ccsc2n1 c1(NC(C23CC(C(N(CC=C)CC=C)=O)(C2)C3)=O)c(Cl)c(F)nc(F)c1Cl c1(C(=O)NCC2(O)CCCN(C(COCC)=O)C2)ccnc2c(Cl)c(C)ccc12 N1(CC)CCC(NC(=O)CCOCCN(C(=O)Cc2ccc(O)cn2)C)CC1 N1(C(Cc2ccc(C)c(O)c2)=O)CC(C)C(NC(=O)C=Cc2cccs2)C(C)C1 N1(C(C=C(C)Cl)=O)CC(NC(=O)C(c2cccc(C(F)(F)F)c2)O)CCC1C Cc1ncnc(N2CCCOC(CNC(=O)C=CC=C(Cl)Cl)C2)c1C#N c1(C(N2CC3(C2)C(=O)N3)=O)cc2ncccc2[nH]1.c1(OCC)cnc(F)nc1 c1(CC(=O)NC(C)CNC(=O)CS(N)(=O)=O)ccccc1S(C)=O C(=O)(CCC(=O)NC(C)CNC(C1C(C(C)(C)Sc2ccccc2)C1)=O)OC n1(CCC2CC(NC(CSCCOCOC)=O)C2)cc(-c2cnccn2)nn1 CCCC(CC)CC(=O)N1CCCCC1CNC(=O)CNC(=O)CC(C)C Cc1ccc(C=CC(N2C(CNC(=O)C(C)NC=O)CC3CCCC23)=O)cc1C C#Cc1cc(C(=O)NC2CC(N(C(=O)CCC3CC3(C)C)C)C2)cc(F)c1 C(CC(C)C(=O)N(CC)CC1CN(C(=O)CCC=CCCC)CCO1)=CCC C1(NC(c2c(CC)[nH]cc2)=O)(COC)CCN(C(c2cnc(Cl)cc2Cl)=O)CC1 c1(CC(=O)NC(C2CCCN2C(=O)Cn2nccc2N)C)ccc2c(c1)CCC2 C1(CNC(C(CSC)C)=O)CCC(C(=O)N(C)Cc2csnc2C)CC1 CCC(C)(C)CC(=O)N1CCC(C(=O)NCC2CC23CC3(F)F)(CC)C1 c1(C(N(CCCOCCN(C(=O)CSCC(F)F)C)C)=O)cc[nH]c(=N)c1 N1(C(CSCC(N)=O)=O)CC2CCOC2(CNC(=O)Cc2cnsc2)C1 Cc1cc(C(N2CCC(F)(F)C(NC(=O)CCCCCO)C2)=O)c(F)c(Br)c1 CC1(CNC2CCC(NC(=O)CNC(N3CCCC3)=O)CC2)CCCCC1 C12(C(=O)NC(C)CN3CCOCC3)CCCC1CCN2C(c1cncc(Cl)c1)=O c1(C(C)N(C(CC=CCC)=O)C(C)C)ccc(NC(C)=O)cc1 c1(C(=O)NCC(N2CC(CCNC(CCSC)=O)C2)=O)c(F)cccc1F CSC1=C(C(=O)NCCCNC(C2CCC2C(F)(F)F)=O)CCCC1 C1(CNC(C(C)O)=O)(NC(c2cccc(C3CN(C)C3)c2)=O)CCOCC1 CC(C)CS(=O)(=O)CC(=O)N1CC(n2cc(CNC(=O)C(C)(C)F)nn2)C1 N1(C(C(c2cccc(Cl)c2)C)=O)CCC2(CC1)CN(C(=O)CC1(CO)CCC1)C2 C#CCC(C(=O)N1CCC1CC(C)C)NC(=O)CN1CCSCC1 c1(C(N(CCCNC(=O)CC(C)(C)COC)CC)=O)cc2occ(Br)c2[nH]1 c1(NC(=O)CC2CCCN2C(=O)C(c2ccc(Cl)cc2)CO)cnnc(O)c1Cl c1(OC)cc(Nc2cccc(C)c2C)ccc1C(c1nnnn1CCSC)OC Cc1cc(=NC(=O)C(=O)NC23CC2CN(C(=O)C#CC2CCCCCC2)C3)[nH]o1 C1(C(=O)NC2CCCC2C)(CC)CCCN(C(=O)CCC(C)(C)N(C)C)C1 C=C(C)CCC(C)NC(=O)C(=O)NC1CCN(CC(=O)O)C1=O C(=O)(CCCCC(F)(F)F)NC1CN(C(c2cccc(NC(N)=O)c2)=O)C1 N1(C(CCNC(CC(C)C)=O)=O)CC(NC(C2CCCN2C=O)=O)CC(F)C1 c1(C(=O)NC(CC(=O)Nc2ccc(OC)nc2)C2CC2)n[nH]c2c1CCC2C N1(C(c2cn(CC)nc2C)=O)CC(CNC(=O)CC2CCOC2)C(F)(F)C1 N1(CC(=O)NCC(CN(C(C2CCC(C(=O)OC)C2)=O)C2CC2)F)CCC(C)(C)C1 C(C)(C(CC(=O)NCc1cn(C(C)C)nn1)NC(=O)Cn1ccnc1)OC C(C1=CCN(C(C2CCN(S(C)(=O)=O)C2)=O)CC1)NC(c1c(CCC)occ1)=O C#Cc1cc(C(N2CCN(C(c3cccc(CC)c3)=O)CC2CO)=O)cc(F)c1 c1(CC)ccc(C(=O)NCC2CC(NC(=O)C=CCCC=C(C)C)CCO2)c(N)c1 C(=O)(CCC(C(=O)NC(C)C(=O)OC)N1CC=CC(N(C)C)C1)OC S(=O)(=O)(c1ccc(C(=O)NCC2CN(C(c3nccn3C)=O)C3CC23)cc1)NC c1(C(=O)NCCCC(CCC)NC(=O)CC=CC(C)(C)C)csc2ccccc12 C1(NC(N(C)Cc2cc(Cl)c(OC(F)F)cc2Cl)=O)CCC(F)(F)CC1(C)C N1(C(c2c(C)cns2)=O)CC(NC(=O)CC2CCCCC23CC3)C(C2CC2)C1 C(CC(=O)NCC(O)CNC(N)=O)(C(C)OC)NC(c1c(CC)non1)=O N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(c2ccco2)=O)CC12CCC2 c1(C(=O)NC2CN(C(=O)C(O)CN3CCCC3)CC2C2CC2)ccc2cc[nH]c2c1 c1(OC)cnnc(C(N2CC(NC(c3cc(SC)c(C)o3)=O)C2)=O)c1 n1(CC(=O)N(CCNC(=O)CCC2CC2C)CC)nc2n(c(=O)c1=O)CCOC2 C(=O)(C(CN(C)C)C(C)C)NC1(CNC(c2sccc2OC)=O)CC(OC)C1 C(=O)(C1=CS(=O)CCC1)NCC(CNC(=O)CCCc1cnccn1)OC Cc1cc(C(=O)NCC2CCC(C)CN2C(=O)Cc2cnsc2)cnc1C(F)F C(=O)(CC1OCc2ccccc21)NC(C)C(C)(C)NC(=O)Cn1ncn(C)c1=O Cc1ncc(C=CC(=O)NCC(C)(O)CNC(c2cccc(F)c2F)=O)c(O)n1 N1(C(CC2(N(C)C)CCC2)=O)CC2CCCN(C(C3CCCN3C=O)=O)C2C1 N1(C(C(c2ccn(C)c2)C)=O)CC2CC(C1)CN(C(C1OCCC1C(C)C)=O)C2 C1(CCCC(C2CSCC(=O)N2)=O)CC2CCC1C2.c1(C(=O)OC)cn(C2CC2)nn1 C#Cc1ccc(N=c2scc(-c3cnnn3C)n2Cc2nn(C)cc2Br)cc1 C1(CC(N2CC(C)(NC(C3N(C(CCC)=O)CSC3)=O)C2)=O)CCC(=O)N1C c1(C(N(C2CCN(C(C3CCCC(C)(C)O3)=O)C2)CC)=O)coc2c1CCCC2 C1(CCNC(CC(C)OC)=O)CCCN(c2ncnc(=N)[nH]2)CC1 c1(-c2scc(C)c2)ccc2c(c1)CN(C(=O)N=c1cccn[nH]1)CC2 c1(CC(C)C)cc(C(N2CC(CNC(c3nccs3)=O)CC2C)=O)cc(O)n1 c1(OC)cccc2c(CNC(c3cc(=O)n(C)cc3Br)=O)csc12 c1(C(=O)NC(C(C)c2ccccc2)CO)cc2c(F)ccc(F)c2s1 Cc1cc2sc(C(N3CCCCC3CN(C(=O)C(F)C(C)C)C)=O)cc2s1 Cc1cccc2[nH]cc(CCC(=O)NCC(O)CNC(c3cnc(S)n3C)=O)c12 Cc1ccc(SCC(=O)NC2CN(C(=O)CC(C)CF)CC2C(F)(F)F)cc1 C(CCC(=O)NC1(C=CC(=O)NOCCF)CCC1)N(C)C CCCCC(C)(F)C(=O)NCC1CC1C(=O)Nc1cc(O)ccc1OC C#Cc1cc(C(N2CC(C(=O)NC(c3ncc(C)s3)C)CCC2C)=O)ccc1C N1(C(C(C)C)=O)CCCC1C(=O)NCCC(C)(C)NC(=O)CCn1ccnc1 C1(C(=O)NC(C(=O)NC(C=C)(C)C)C)Cc2nccn2C1 CC(C)CC(C(=O)N1CC2CC2(CNC(=O)C=Cc2ccco2)C1)C(N)=O C1(NC(C(Br)=C(C)C)=O)CC(C)N(C(c2coc(-c3ccccc3)n2)=O)C1 CC1CS(=O)(=O)CCCN1C(C(=O)NCCC#N)C1CC1Cc1nnn(C)n1 CCCC(C(=O)NC1C2COCC12)NC(c1n[nH]c(C)c1O)=O C(=O)(CCCCCCCNC(C)=O)N1CCN(c2c(F)cc(OC)cc2F)CC1 C1(C(=O)NC2C(CNC(c3[nH]cc(C(C)=O)c3)=O)CCC2)CCCCCCC1 c1(C(N2CC(C#C)(C(=O)NC3(C)CCSC3)C2)=O)ccc2cncn2c1 c1(C(N2CC3C(CNC(C(C)(C)F)=O)(C3)C2)=O)c(O)cnc2ccccc12 C(=O)(CCCCCNC(N)=O)NCC(C(C)(C)C)NC(CN(C1CCSC1)C)=O N1(C(c2scc(CNC(CCN(CCC)C)=O)c2)=O)CCC(C2CCOC2)C1 N=c1ccc(C(=O)NCCOCCNC(C2CC2c2cccc(Cl)c2)=O)n[nH]1 C1(OC)CC(CC(C)(C)C)CN(C(=O)C(C)CC(N)=O)C1.C(=O)CC(=O)N(C(=O)CN)C CCCC(C(=O)NCCCCCC(=O)NCC1(C)CCC(=O)N1)C(C)C C1(CNC(=O)Cn2nccn2)C2CCC(C2)N1C(c1ncccc1C1CC1)=O CC1(C)CCC(O)(C(=O)NC2CC3CN(c4nccn5nnnc45)CC3C2)CC1 N1(C(C2CC(CCC)OCC2)=O)CCOC(C)(CNC(c2cc(F)n(C)n2)=O)C1 C1(C(=O)NC(CC2CCN(C(CN(CCC)C)=O)CC2)C)CCCC12OCCO2 c1(C(N2CCS(=O)C(C)C2)C(=O)NCC)cc(Cl)c(Cl)c(Cl)c1 N1(C(c2ccc(C)nc2O)=O)CCCC2(NC(C3CCC(F)C3)=O)CC2C1 c1(CCC(=O)N(CC(CC)NC(C(C)OCCC=C)=O)C)ccccc1OC C12(CNC(c3cnc(C)s3)=O)CC(CN1C(c1cocn1)=O)C2 N1(C(c2cn(CC)nn2)=O)CC(C)OC2(CCN(C(=O)C(CO)N(C)C)CC2)C1 c1(C(N(C2CCCN(C(=O)C(C)(C)F)C2)CC)=O)cccc(C)c1N N(C1CCCc2c1cnn2C)C(C1CCN(C(=O)OC(C)(C)C)CC1C(=O)O)=O C1(CCN(C(c2c(C)nns2)=O)C)CCN(C(=O)CSC(C)(C)C)CC1 CSC1=C(C(=O)N2CCC(NC(c3cnn4ccsc34)=O)C2)CCCC1 c1(C(=O)NC2CC(C)(CNC(=O)Cn3cnnc3)C2)ccc(F)cn1 c1(C(N2CC(O)(CNC(C3(CN(C)C)CC3)=O)C2)=O)cc2nccc(Cl)c2s1 C1(C#N)(C(N2CCN(C(C(C)CC3CC3)=O)CC2)=O)CC2(CC2)C1 C(=O)(CCCS(C)(=O)=O)N1CCC(C)C1CNC(c1cc(=O)n(C)o1)=O C(C(=O)NC(C(=O)NCc1ccc(C)o1)C1CCC1)(C(C)(C)C)OC C1(CNC(C2CCCC2C(F)F)=O)CC(F)(F)CN1C(=O)Cc1ccnc(F)c1 C(CC(C)(CC)NC(=O)CCCF)NC(c1ccc(CC)o1)=O CCCC(O)(CCC)CC(=O)NCCCN(C)C(c1ccc(OC(C)C)cc1)=O N1(Cc2nnn(C)n2)C2CCC1CN(C(c1cnc(C3CCC3)nc1O)=O)CC2 c1(CC)cc(C(N2CCC(CN(C)C(C3NC(=O)OC3C)=O)C2)=O)cc(Cl)c1 S(=O)(=O)(CCN=C(NCc1ccc(C)o1)NCc1ccc(OC(F)F)cc1)NC c1(C(=O)NC(C2CN(C(c3cc4c(ncn4C)s3)=O)C2)C)csc2cccnc12 c1(C(N2C3CN(C(C4COCCO4)=O)CC2CC3)=O)cc2ccccc2nn1 Cc1ncc(N)cc1C(=O)NC(C1CCCC1)CNC(c1nncn1C)=O Cc1c(C(N2CCN(C(=O)Cc3cncc(C#N)c3)CC2)=O)nn2c1OCCC2 C1(CNC(C2(CC)COC2)=O)CC2(CC2)CN1C(=O)Cn1cnnn1 C1(C(N(C2CCN(C(C3(CC=C)CC3)=O)C2)CC)=O)CCC(F)(F)CC1 N1(C(c2c(C#N)nc(C)o2)=O)Cc2[nH]nc(NC(c3cccc(Cl)c3Cl)=O)c2C1 CC1CN(C(=O)CCOCC(F)F)CC1NC(c1cccc(CF)c1)=O Cc1ccc(CN2CCCC(C)(C(=O)NOC3CC4CCC3C4)C2)c2c1CCC2 CCCC(CC)C(=O)NC1CCN(CCNC(C2CC(C)OC(C)C2)=O)CC1 Cc1cccc(C(=O)NCC2CC(CC(=O)NC3(C)CCCCCC3)C2)c1O C12(NC(C3C(C(C)C)C3)=O)CCC(CC1n1cc(COCC(C)O)nn1)C2 CC(C)CC(CO)CN=c1ccc(S(=O)(=O)NC(C(C)(C)C)C2CCC2)c[nH]1 C(CCCCOC(N)=O)N(c1cn(CCNS(N)(=O)=O)nn1)C(C)(C)C O=S(=O)(c1ccc(N2CC(O)CC(O)C2)c(Cl)c1)NCc1csc(C(F)F)n1 Cc1ccccc1C1=NOC(C(N2CCOC(CNC(C3(Cl)CC3)=O)C2)=O)C1 C=CC1(C(=O)NCCC2CN(C(C3CC(C)(C)CO3)=O)CCO2)CCCCC1 Cc1c(C(=O)NC2CC=CCC2C(=O)Nn2ccnn2)cccc1C#N N1(C(C)=O)CCCC1(C)C(=O)NC1CC(N(C(=O)Cc2cc(C(C)C)no2)C)C1 c1(C(=O)NC2(C)CCN(c3ncc(C)cn3)CC2)c(C)nc2sccn12 C(c1ccc(F)c(F)c1)=CC(=O)NC1C2CN(C(C=CC(C)C)=O)C1C2 C1(C(N2CCC(CC)C2CNC(C2CCOC2(C)C)=O)=O)CCCCCCC1 c1(OC)cc(CO)ccc1C(=O)N(CC(O)CNC(C1CCO1)=O)C C1(NC(CC2(CC)CC2)=O)CCN(C(=O)COCc2ccnn2C)C12CCC2 c1(OC(=O)OCC)ccc(C)cc1CNC(c1ccccc1F)=O C1(C(N(C)CC2CCN(C)C2)=O)CCCCCCN1C(=O)CC1(O)CCOC1 C1(NC(COCCC)=O)CCN(C(c2ccn(C(C)C)n2)=O)CC1C Cc1n[nH]c(C)c1C(=O)NC(CO)C(C)NC(C1CC(F)C1)=O N1(C(c2c(SC)scc2)=O)CC2OCC(NC(c3coc(Cl)n3)=O)C2C1 c1(C(C)=O)cccc(OCC(N2CCCC(NC(c3cc(Cl)cs3)=O)C2)=O)c1 C1(C(C)C)(NC(C2CC(OC(C)C)C2)=O)CCN(C(=O)C(F)CC2CCOC2)C1 C1(CCC(=O)N(C(C)(C(=O)NC2(C(C)O)CC2)C2CC2)C)NC(=O)NC1=O C1(CC(=O)NCC(CCOC)NC(c2ccn(C)c(=O)c2)=O)CCCC(C)(C)O1 C1(CC(=O)NC(CNC(c2cnc(CC)[nH]2)=O)CC)CCCC(F)(F)C1 N1(C(C(C)CF)=O)CC(CNC(=O)COc2cccc(Br)c2)CC(C)(C)C1 c1(CC(N2CC3CC(NC(=O)COC4CC4)C3C2)=O)ccc2c(c1)CCCC2 c1(C(=O)NC2CC(F)(CNC(c3cnc4n3CCC4)=O)C2)cccc2c[nH]nc12 C1(C)(NC(C(CO)OC)=O)CCCN(C(c2cncc(F)c2)=O)C1 S(=O)(=O)(c1cccnc1)N1CC(C(=O)NCC2CCCC2)OCC1 C1(CC(=O)NCCCCC(=O)NC2CCCC2(F)F)CCCNC1=O c1(C(N2C(CN(C(=O)CC3CC3(C)C)C)CCC2)=O)cc2ccncc2[nH]1 c1(C(=O)NC2C(SC)CCC2)ccc(CNC(c2ccoc2Cl)=O)nc1 N1(C(C2CC(NCc3c(F)cc(I)cc3F)C2)=O)CCc2cccc(Br)c2C1 n1(CCNC2C(S(C)(=O)=O)CCCC2)cnc2ccccc2c1=O N1(C(=O)Nc2ncc(CS(=O)(=O)c3ccccc3)s2)Cc2cccc(CO)c2C1 Nc1cccc(C(=O)NCCCNC(C2CC(F)(CF)C2)=O)c1F N1(C(COCCC=C)=O)CCC(C=CC(N2CC(CO)OCC2C)=O)CC1 C(C(O)CC(=O)NCC(C)(C)C1CC1)NC(c1nc(CCC)oc1)=O C1(NC(CC=C)=O)CC12CCN(C(C1CC=CCN1C(=O)OC(C)(C)C)=O)CC2 C(=O)(CCC(=O)NCC1CCCC1)NCC.c12ccccc1CNC(=O)C2(F)F c1(OC)cc(Br)c(Cl)cc1C(=O)NC(Cc1ccccc1)C(C)c1ccccc1 N1(CC)CCOC(C(=O)NC(c2nc(C)c(CNC(=O)COC(=O)C3CC3)s2)C)C1.CC C1(C(N2CCC(C)(CN(CC(F)(F)F)C)C2)=O)C2CN(S(C)(=O)=O)CC12 C1(CC(=O)NC2CC(C)(NC(C3C(C)(C)CC3)=O)C2)Cc2ccccc2NC1=O CN1C(=O)CC(c2nc(-c3cccc(Cl)c3)nn2Cc2ccsc2)NC1=O n1(CC)ccc(C(=O)NCC2CN(C(=O)C(C)(C)C#N)CCO2)cc1=O N1(C(c2c(C)ccc(Br)c2)=O)CCOC2(CCCN(Cc3cc(Cl)sc3Cl)C2)C1 C1(CCNC(c2cc(CCC)[nH]n2)=O)NC(=O)NC1=O.C1C(C)=CC(=O)N1 C1(NC(c2cccc(O)n2)=O)CCC2(CC1)CCN(C(c1cccnc1O)=O)C2 C1(NC(C2N(C(C3C(C)(CC)C3)=O)CCC2)=O)CCCC2(C1)N=N2 c1(C(=O)NCCN(C(C2CC2OC(C)=O)=O)CC)sc(C)nc1C C1(CNC(CCCCC)=O)CCC2CN(C(c3nn(C)cc3C)=O)CC12 c1(CNC(C(=O)Nc2cccc(C(=O)NC(C)=O)c2C)=O)cc(C)cc(C)c1O Cc1cc(C(=O)NC2CCN(C(c3n[nH]cc3Cl)=O)C23CCC3)n2ncnc2n1 C1(C(=O)NCCN(C(c2c(C(C)C)c[nH]n2)=O)C)Cc2cscc2C1 C1(CC)COCCN(C(=O)Cc2ccc(C(C)C(F)(F)F)cc2)C1 C(=O)(C(C)CC(C)(C)C)NCCCC(CCC)NC(c1ccc(C#N)nc1O)=O C(=O)(C(CCC(N)=O)N(C)C)N1C(CNC(Cc2c(C)ccc(C)c2)=O)CCC1 c1(C(N2C(C)CCC2C(=O)NC(C#N)C(N)=O)=O)cccc2cc(Br)cnc12 C1(O)(CNC(c2n(C(C)C)ccc2)=O)CCCN(C(c2scnc2Cl)=O)C1 c1(OC(C)C)ccc2c(c1)CCCC2NCC1(O)CC2CCC(C1)N2C c1(C(=O)OC)cnn2c1CN(C1CCCN(CC(=O)OC)C1=O)CC2 N1(C(CC(=O)OCC)=O)CCC2C(C1)CN2C(=O)CC(C)n1ccnc1C(=O)OC C(=O)(CCCCCS(N)(=O)=O)NC(C(C)NC(C(C)SCC)=O)C c1(C2C(SCC(=O)NC3CC(N(C(C(C)=C4CCC4)=O)C)C3)C2)ccccc1 C1CCCC(=O)N1.C1(CNC(N)=O)CCC(C(N2CC(NC(N)=O)C2)=O)C1 N1(C(CCC=C)=O)CCC(NC(=O)CCN2CCCC2=O)C(O)C1 C(=O)(CCCCCO)N1CCCC(N(C(CCc2ccc(C)cc2)=O)CCO)C1 N1(C(CCCNC(C(C(C)C)F)=O)=O)CCN2CC(O)CC2C1 C1(C(=O)NCC2C(NC(COCCCC)=O)C2)CCC2(CCC2)CC1 c1(C(=O)NC(C)C(C)NC(=O)CC#N)ccc(C(=O)C(C)(C)C)cc1 C(=O)(C(C)C1=CCCC1)NC(C(C)C)CNC(=O)C=Cc1ncco1 c1(NCC2N(C)CC(O)CC2)c(F)cc([N+](=O)[O-])cc1F C(CC(C)(C)C(=O)NC(CNC(c1cc(F)cnc1OC)=O)CO)OC C1(C(=O)NCCN(C(=O)Cc2ccccc2F)C2CC2)OC2CCC1C2 c1(C(=O)NCCSc2onc(CCNC(=O)Cn3ccnc3)n2)cnnc(O)c1 N1(C(C(C=C)c2ccccc2)=O)CCN(C(=O)Cc2cnn(C)c2C)CC1CC O=C(C1CCCCc2ccccc21)NC1C2CN(C(=O)C(F)=CC3CC3)CC12 CC1(C(N2CC(CNC(=O)CCc3cc(Cl)no3)C(O)C2)=O)CCC(=O)N1 c1(C(=O)OC)cc(F)cc2c1CN(N1CC=CC1C(=O)OC(C)C)CC2 C(=O)(C1=NOC(CNC(C2CCC(=O)C2)=O)C1)N(CC(=O)NCC1CC1)C C(CCO)(C(=O)NC1CCCN(C(=O)C(C)(C)n2cnnn2)C1)N(C)C C1(C(N(C(C)CNC(=O)C(C)(C)N2CCCC2)C)=O)CC(=O)N(C)C1 CC(O)C(C(=O)N1CCN(CC2CN(C(C3CC=CCC3)=O)C2)CC1)OC.CCO N1(C(C2N(C(C3C(=C)C3C(=O)OC)=O)CCC2)=O)CC(=O)N(C)CC1C N1(C(c2c(CC)nns2)=O)CCC2(CC1)CN(C(C1CCC1)=O)CC(C)O2 c1(SC)ccc(O)c(C(=O)NCC2CCCCN2C(C2CCCCS2(=O)=O)=O)c1 C=CC1(C(=O)NC(C)Cc2cnn(C)c2)CCN(C(C2CCCCO2)=O)CC1 C(C1c2ccccc2CCN1C(=O)CSC1CCCCC1)NC(C(C)OCC)=O O=C(C#CC1CCCCC1)NC1CN(C(C2CC3CCC(C2)O3)=O)C1 CCCCS(=O)(=O)CC(=O)N1CCOC2CN(C(c3ccsc3C#N)=O)CC12 c1(CC(N2CC(CNC(C(F)=CC)=O)C(C(N)=O)C2)=O)ccc(Cl)c(OC)c1 C1(N(C(C2ON=C(C)C2)=O)C)CCN(C(=O)C(C2CCCCCC2)F)CC1 Cc1nn[nH]c1C(N1CCC(N(C(=O)Cc2cnc(C3CC3)[nH]2)C)C1)=O CC1CCN(C(c2cnc(-c3ccccc3)s2)=O)C1CNC(=O)CCC(C)O CC(C(=O)NCC(C(C)(C)C)NC(c1ccncn1)=O)C(C)(C)O CC1CN(C(=O)C=CC2CCCN2C(=O)Cc2cccc(C3CC3)c2)CCS1 C1(C(N2C3CN(C(CCP(C)(C)=O)=O)C(C3)C2)=O)C2CCCCCCC12 c1(-c2nc(CC(C)OC)nn2-c2cnnn2C)ccc(OC)c(SC)c1 N1(C(CCOC(C)C)=O)CC(NC(c2ccn(C(C)C)n2)=O)CC12CCCCC2 c1(C(N2CCN(CCNC(C34CCC(C3)C4)=O)CC2)=O)ccnc2[nH]cnc12 c1(CC)cc2c(CC(=O)NCC3CCC(NC(=O)C4=C(Cl)CCC4)C3)csc2s1 c1(C(N2C(C)CC(NC(=O)Cn3ccnn3)CC2)=O)noc2ccccc12 c1(CC)nc(C)c(CC(=O)NC2CS(=O)(=O)CC2NC(=O)C=CCF)c(C)n1 C(=O)(CC(CC)C(F)F)NCCC1(O)CN(C(C2CC(OCC)C2)=O)C1 N1(C(CC2CCN(C(C(C)(C)C3CCCO3)=O)CC2)=O)CCC(O)C(O)C1 c1(CC)nn(C)c(C(N2CC3C(NC(=O)C(C)(C)Cl)C3C2)=O)c1Cl C=CCCC(F)(F)C(=O)NCCCC1(NC(=O)C=Cc2cnn(C)c2)CC1 N1(C(CSCC(=O)OC)=O)CC(CNC(C2(OC)CC2)=O)OC2CCCC12 c1(C(N2CC(C#C)(C(=O)NC(C3CC3C(N)=O)C)C2)=O)cc2ccccc2o1 O=C(C(Cl)=CCl)NC(CNC(=O)Cc1cc(C2CCC2)no1)C1CC1 Cn1ncc2c(CCNC(=O)CNC(C3CC(=O)N(C)CCN3)=O)ncnc12 c1(CC(=O)NCC2(NC(C3(OC(C)=O)CC3)=O)CCC2)csc(Cl)n1 C1(C(N2Cc3c[nH]nc3C2)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(F)F C#Cc1ccc(Cl)c(C(=O)NC2CCCN(C(c3cccnn3)=O)CC2F)c1 CC1(F)CCCN(C(=O)C(CC(F)F)NC(=O)CN2CCOCC2=O)C1 C(=O)(C1CCOc2ccc(Cl)cc21)NC1C(NC(=O)Cc2ccon2)C1 C1(=C(C(=O)NCC(CNC(C(C)=CC)=O)C)F)CCCCC1 c1(C(c2nnnn2CCCF)NC(c2nc(CO)co2)C)ncoc1C(F)(F)F C#CC1COCCN1C(C1CC2CC2N1C(=O)C(CC(=C)C)OC)=O N1(CCCC)CCOCC1C(N1CCC(C(C)NC(=O)OC(C)(C)C)CC1)=O c1(OC)cccc(OC)c1CC(N1CC2CC1C2CNC(C1(Br)CC1)=O)=O C(=O)(C(F)C(C)(C)O)N1CCCC(C(C)NC(=O)CN2CCOCC2=O)C1 C(CS(=O)(=O)CC)NC(c1n(CCCSCC)nnn1)c1cnc(CCOC)s1 C1(COC)CC(NC(C2(C#C)CCC2)=O)CN1C(c1ccnc(OC)c1)=O N1(C(C(N2CCOC(C3CC3)C2)C)=O)CCCCC(NC(=O)C2CC2)C1 c1(C(=O)NC(CCCC)COC)c[nH]cc(C)c1=O c1(C(N2CC(CCNC(C3(SC)CC3)=O)C(C)C2)=O)cc2cc(OC)ccc2[nH]1 N1(C(c2ccc(COC)[nH]2)=O)CC(CNC(C2CCC2)=O)C(O)C1 N1(C(C)C(=O)NCC(c2nccs2)C)CCN(CCCC#N)CC1 C1(C)(CC)CC(NC(=O)CCSc2cccc(F)c2)CN1C(=O)C(F)=C1CCC1 C(=O)(CCCCCCBr)N1CCC(C(C)NC(=O)Cc2ccnc(Br)c2)CC1 C(=O)(C(F)C(C)CNC(=O)C(C)n1cccn1)N1CC(CCC#C)C1 N1(C(c2c(Cl)ccc(C)c2)=O)CCN(C(c2ccc(Br)c(C)c2)=O)CC1C#N N1(C(CS(=O)(=O)NC)=O)CCOC2CN(C(=O)CNC(C3CCOCC3)=O)CC12 c1(C(=O)NC(C2CCN(C(c3cccnc3O)=O)C2)C)c(Cl)ccnc1F c1(C(=O)NC2(CC)CCN(C(C34CC(C3)C4)=O)CC2)ccc(F)c(F)c1F N1(C(C2C(CCOC)C2)=O)CC(=O)CC1C(=O)NCC(C)(CC)CC C(CC(C(=O)OC)NC1COC1=O)=CC.C(c1c[nH]cn1)=CC C1(OC)(CNC(=O)C(F)(F)C2(OC)CCCC2)CCN(C(=O)C(O)C(C)C)C1 N1(C(c2cn(C)nc2)=O)CCN(C(C2CC2(C)C)=O)CC1C1CC1 Cc1sc(C(N2CCCC2CN(C(=O)CC2CCSC2)C2CC2)=O)nc1O CCC(CCC(=O)NCCC1(CO)CCCC1)NC(C1CCNC1=O)=O Cc1snnc1C(=O)NC(C)C(C)(C)NC(=O)C(CO)c1ccccc1 C(C(C(=O)NCC(CO)NC(=O)CN(C)C(=O)O)NC1CC1)OC.C(C)(C)(C)O CC(C)CCC(F)C(=O)N1CC=C(CNC(=O)C(C)S(C)(=O)=O)CC1 N1(C(Cn2ncc(C)cc2=O)=O)CCOCC(C)(CNC(=O)CC2CCCO2)C1 N1(C(C(COC)(C)C)=O)CCC2(CCCN(C(C3CN(CP(C)(C)=O)C3)=O)C2)C1 Nc1cc(C(=O)NC2CCCN(C(c3occc3Cl)=O)CC2)cc(F)c1O C12(C(=O)NC(CNC(C(CC)CCOC)=O)C)CC3CC(C1)C(F)(F)C(C3)C2 CC(C)CC(CNC(C1CN(C)C(=O)N1)=O)C(=O)NCCc1cnccn1 O=C(C1=CC2(CCOCC2)C1)NCC1CC1NC(=O)Cn1cc([N+](=O)[O-])cn1 C1(OCC(=O)NCC(C2CCCC2)NC(c2ccc[nH]2)=O)CC=CC1 C1(C(N2CCC(C(C(=O)NC3C(C)CN(C)C3)(C)C)C2)=O)CC2(C1)CC21CC1 CC1CCC2(CC1)CCC(COC(c1cnn3ncccc13)=O)O2 c1(CC(CNC(C(C)N(C(=O)C=O)CC)=O)O)ccc(O)cc1.C(C)(C)(C)OC(=O)N CC1CCN(C(c2cocn2)=O)CCN1C(c1ccn2cncc2c1)=O CC1(C)CC(C(=O)NCCC2(C(N3CC(CO)C3(C)C)=O)CC2)CCO1 c1(C(N2CC(C(C(=O)NCc3cnco3)OC)C2)=O)cccc[n+]1[O-] Cc1cc(Cl)ncc1CC(N1CCN(C(=O)CCc2ccc(=N)[nH]c2)C2CC12)=O C(CCCCCN(C)C(c1cc(CC)cn1C)=O)NC(C1(CC#C)CC1)=O N1(C(c2c(C)cc[nH]2)=O)CC2CC(NC(c3ccccc3NC(N)=O)=O)CC1C2 C12CCC(C)(C1)N2.C1(CC(=O)C2CC2)(COC)CCC1.c1(CC(=O)NC)ccon1.S c1(OC)cc(NC(C2(C)CCN2C(=O)C(C)c2cccs2)=O)cc(OC)n1 Cc1cnc(OCCNC(C2(c3ccccc3)CCCC2C)=O)c(C)n1 CCCC(C(O)C(=O)NC(CO)C(=O)OC)NC(=O)CCCN(C(N)=O)C C(CC(C)C)(C(=O)NC1CC(CO)C12CCC2)NC(c1c(C)ncnc1)=O Cn1ccc(-c2cn(CCCC(=O)NCC3C4CCCC34)nn2)cc1=O C12(CCN(C(=O)CN3CC(=O)NC3=O)CC1)CC(=O)N2.c1(CC)nnccc1C CC1CCN(C(=O)CCn2ccccc2=O)CC1N(C(=O)CC1CCSCC1)C N1(N2C(CNC(C3C(C4CC4)C3(F)F)=O)CC(F)C2)CCC(F)CC1.C=O c1(C(=O)NC(C(CO)NC(c2n(C)nc(C)c2Cl)=O)C)csc2c(O)ccnc12 Cc1cc(C(=O)NCC2CN(C)CCN2C(C2C3CC4C(C3)C24)=O)nc(Cl)c1 C1(C(=O)NCCCNC(C2(C#N)CC(C)C2)=O)CCOC2(CCC2)C1 N1(C(CC(C)C(C)(C)C)=O)CC2(CCN(C(=O)C=Cc3ccccc3)CC2)C1 C1(C(N(C)Cc2ccco2)=O)CCOCCN1C(=O)CCN=[N+]=[N-] C(=O)(C1=CCOCC1)N1C(CCNC(C(C)CN(C)C)=O)CCCC1 Cc1ncccc1C(N1CCC(C(=O)N(CC(C)O)C)(N(C)C)C1)=O C1(C(N(CCNC(c2cncc(OC(F)(F)F)c2)=O)CC)=O)CC(F)C(=O)N1C N1(C(C=Cc2cnc(C)s2)=O)CC2(CCC(NC(=O)CSc3nc[nH]n3)C2)C1 C=CC1CN(C(C2OCCC2C(C)C)=O)CC1NC(c1ccnn1CCC)=O c1(C(=O)NC2CC(NC(C3C(C(=O)OC)CC3)=O)C2)nn(C)c(=O)cc1C c1(C(C(=O)NCCCSCC)N(C)CCC2CC2)cccnc1F Cc1ccc(C(=O)NC2COCCC2NC(=O)CCc2cnn[nH]2)cc1F Cn1nc(C2CC2)cc1C(=O)NCCC1CCC(NC(c2ccc(Cl)cn2)=O)C1 N1(C(C(=O)NCC(=C)C)c2cccs2)CCC(O)(c2nc[nH]n2)CC1 c1(CS(N2CC(CN(c3cc(F)cc(Br)c3)C)C2)(=O)=O)ccc(S(C)(=O)=O)cc1 c1(C(=O)NCC2C(C(=O)Nc3c(C)scc3)CCC2)cc(O)cc(F)c1 c1(NC)ncc2c(n1)CCOC2.C1(OC)C(OC)CN2C1C2 c1(C(N2CC(C(C)NC(=O)CCN3CCCC3=O)C2)=O)cncc(F)n1 C(C(=O)N(C)OCc1ccccc1)(C1CCC1)N(C(=O)C(c1ccccc1)F)C N1(NC(C2(C(=O)OC)CC2)=O)Cc2ccc(-c3ccc4nc(O)[nH]c4c3)cc2C1 CC(C)C(C(=O)NC1CCCC1NC=O)c1ccc(Cl)cc1.c1ncccc1I Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC1(NC(=O)C(C)(C)c2cnc[nH]2)CC1 CC1CCSCCN1C(=O)C(C1CC1)NC(=O)CC1CCCC12CC2 C(=O)(C(C)(C)CCF)NC(CNC(C(CCC)OCC)=O)CC N1(C(C2C(C)(CC)C2)=O)CC2(C1)SCCC2NC(=O)C=Cc1ncc[nH]1 n1(C(C)CC(=O)NC2CC(NC(=O)C#CC(C)(C)C)C2)c(=O)oc2ccccc12 c1(CC(=O)NC2C(NC(C(F)OC)=O)C2)ccccc1C C(=O)(CC(C)(C)N(C)C(=O)Nc1cccc(-n2ccnc2)c1)OC N1(C(c2nn(C)cc2Br)C(=O)NCC(=C)C)CC(COC)OC(CC)C1 N1(C(C2=C(C)CCC2)=O)CCCC2(CCCN2C(c2cocc2C)=O)C1 N1(C(C(SC)SC)=O)CCN(C(=O)C(CC)c2ccccc2)C(C2CC2)C1 C(=O)(C1Cc2c(Cl)cccc21)NCCN(C(C(N1CCCCC1)C)=O)CC1CC1 Cc1cnc(C(N2CC3C(NC(c4cc(C(C)C)ccc4C)=O)C3C2)=O)c(F)c1 C(=O)(CCC(=O)N1CCCC1C(C)(C)NC(C1(C)CCOC1)=O)c1ccc(C)s1 c1(OC2C(C(=O)NC3(CC=C)CN(C(=O)C(N)=O)C3)C2)ccc(SC)c(Cl)c1 c1(NOC(c2cccc(CCC)c2)=O)ccc(-c2ccccc2COC)cc1F c1(C(N2CC(NC(C(CC)C#N)=O)C(OC)C2)=O)cn(C)c(=O)n1C C(=O)(C1=NNC(=O)CC1)NC1CC(CCNC(c2c(C)n(C3CC3)nc2)=O)C1 N1(C(CC(CCC)C)=O)CCN(C(=O)C(=CC2CCCC2)C)CC(O)C1 S(=O)(=O)(c1ccc(C#N)c(NCC2(C)CC(F)(F)C2)c1)NCC1(CC)CCC1 N1(C(CCC(C)(C)C)=O)CC2OCCN(C(=O)C(=O)NCCOC(C)(C)C)C2C1 C(N=c1ccn(C(N2CCC2)=O)c(O)n1)c1c(OC)cc(F)cc1 Cc1ccc(F)c(C(=O)NC2(C#N)CCN(Cc3c(Br)ccc(Cl)c3F)C2)c1Br N1(C(c2nc(CCCCC)sc2)=O)CCN(C(C2CCC(C(N)=O)O2)=O)CC1 C1(C(=O)NC(C(=O)NC(c2cn[nH]c2)C)CC2CC2)C2CCCOC12 C(N=c1[nH]c(=NCCN2CCOCC2)[nH]c2c1CSC2)C1(C(F)(F)F)CC1 C=C(C)CCCC(=O)N(CCNC(c1cc(-c2ccc(Cl)cc2)on1)=O)CC N1(C(C2CCC(C)C2)=O)CC2(C(N3CC(c4ccncc4)C3)=O)CC1CCO2 N1(C(C2C(C)(Br)C2)=O)CC2CC(NC(c3ccnc(C4CC4)n3)=O)CC1C2 C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC1CC(NC(=O)C#CC(C)C)C1)C2 C1(C(N2C(NCC3(C)CC3(F)F)CCC2)=O)Cc2c(F)cccc2O1 N1(C(C2(C#C)CCN2C(=O)C2=NOCC2)=O)CCC(C)CC(C)C1 N1(C(c2ccoc2)=O)CCC2(COC(CNC(C34CC(CN3C3CC3)C4)=O)C2)C1 CC(CC1CCC1)C(=O)N1CCC1CNC(=O)CCOCC(F)F CC(C)CC(CC(=O)N1CC(NC(c2sc3ccccc3c2Cl)=O)C1)CC(N)=O C1(COC)CC(C)N(C(=O)CNC(C)=O)C1.N12CCCC1C2=O Cc1c[nH]cc(C(=O)NCC2C(NC(=O)C(C)C)C2)c1=O.C1(=O)CCCN1 CN1CCC(NCC2(CO)CCC2c2ccccc2)C(C)(C)C1 C1(NC(c2cncc(C)c2)=O)COC2(C1)CN(C(=O)Cc1ncncc1Cl)C2 Cc1noc2nc(C3CC3)c(Cl)c(C(=O)NCC3CCCN3C(C3CC3C)=O)c12 Cc1ccc(C(C)C(N2CC(CNC(=O)C=CCF)C(O)C2)=O)cc1 c1(CC(C)N(C(=O)C(C)(C)CF)CC)ccc(CNC(CSCC(C)C)=O)cc1 C(=O)(CCC(C)(C)N(C)CC)N(CCCC(N1CCC(O)(c2cnn[nH]2)C1)=O)C N1(C(COCCOCC)=O)CCC2CCCC12C(=O)NCc1ccc(F)c(Cl)c1 C12(NC(c3ccc(C)s3)=O)CCCC1N(C(=O)C1=CCC(C)CC1)CCC2 C12CC3CC1CN(C3)C(=O)C(C)(C)OC2=O.C1(C)(CC)CN(C(=O)NC)C1 C1(NC(CC2(OCC)CC2)=O)CN(C(c2ccnc(C(N)=O)c2)=O)CC2(CC2)C1 c1(C(=O)NC2CN(C(c3scc(C)c3Cl)=O)C(C)C2)cnc2occc2c1 C1(CNC(c2[nH]cc(OC)c(=O)c2)=O)CN(C(c2cc(C)ns2)=O)C2(CCC2)C1 C1(CNC(C(CN(C)C)NC(C(C(C)C)=O)=O)=O)CCC(C)N1C c1(C(=O)NCC2C(CNC(c3cc(C)sc3C)=O)C2)ccc2c(c1)CCO2 C1(C)(CC)CC(NC(=O)C(C)(C)COC)CN1C(c1cc(OC)ncn1)=O CCC(C)CC(C(=O)NCC1CCC1)NC(=O)C=Cc1cnc(C)s1.C1C(=O)N1 C(N=c1[nH]c(=N)[nH]c(=NC2CCCSCC2)[nH]1)c1nc(CC)sc1 c1(-c2ccc(CNc3nccc(C)n3)cc2F)c2ccccc2nn1C C1(NC(c2cn(CCC)nc2)=O)CCN(C(c2ccc(F)cc2F)=O)C1(C)C N1(C(C2C(C)(C(F)(F)F)C2)=O)CCC(C2CC2)C1CNC(=O)CCc1cn[nH]c1 C1(NC(C(C)CC2CCC2)=O)C2CC3CN(C(=O)CC4CC45CC5)C1C3C2 N1(C(C=CC(C)(C)C)=O)CCOC(CCCNC(C2CC(O)C2)=O)C1 CCCCCCCCCC(=O)N(CC(CC)NC(C1(n2ccnn2)CC1)=O)C C1(C(=O)NC2CC(CNC(c3nc(NC(C)=O)sc3)=O)C2)CCn2ncnc2C1 C12(CC(=O)Nc3c(C)nn(C)c3)CCC1CN(C(=O)CN1CC(=O)NC1=O)C2 C(=O)(C1=CCCOCC1)N1CCC(C)C(CNC(C2CC=CC2)=O)C1 CC(C)CCCCCC(=O)N(CCC(=O)NC(C)CCCCO)CCO c1(N2CCCC(C(C)(C)C)C2)ccc(S(=O)(=O)NC2(C)CCCCC2(F)F)cn1 C1(CNC(=NC)NCCC2(COC)CCCO2)CC(C)(C)CO1 C(C)(C(=O)N1CC2C(NC(c3ccc(N)c(Cl)c3)=O)C2C1)(C(C)C)NC(C)=O C1(CC(F)F)(CC)CCN(C(=O)OCC2CCCCN2C(=O)C(C)=CC2CC2)C1 c1(C(=O)NCC2C(CNC(C(C)OCCOCC)=O)C2)cc(CC)c(=O)n(C)c1 C(=O)(C1=CCC(C)CC1)N1CCC(C(C)C(=O)NC(C)(C)CO)CC1 C=C(Cl)C(C)(C)C(=O)NCCN(C(C12CCC(CC)(C1)OC2)=O)C1CC1 C1(CCCC)CCCN1C(c1ncc(-c2cccs2)s1)C(=O)NC1(C)CC1 c1(OC)ccc(Br)c(C(N2CCC(N(C)C(c3cc(C)cs3)=O)C2)=O)c1F c1(N(CC(=O)NC(c2ccc(OC(F)F)cc2)CCC)C)ncc(Br)c(OC)n1 c1(C(=O)NCc2cccc(NC(CCOCC(C)C)=O)c2)occ2c1CCOC2 CCC(C)CC(C(=O)NC1(C)CCC2(CC1)CC2)NC(c1ccc(F)c(F)c1)=O C1(C(=O)NCC2(COC)CC2)CCOC1CNC(=O)Cc1cc[nH]n1 C1(C(N2CCC(N(C)C)C2)=O)CN(C(C2CCCO2)=O)CC1F c1(OC)cnc(C(N2CC=CC2CNC(=O)COCc2ccncc2)=O)c(F)c1 c1(COC)cc(C(=O)NCCC(C)N(C)C(c2ccn(CC(F)F)n2)=O)n[nH]1 N(C)(C1CCCc2ccccc21)C(c1cc(CC)nn1C)C(=O)NC1COC1 N1(CCC(=O)NC2CC(CCNC(=O)Cn3nccn3)C2)CCOCC1=O C1(CCNC(Cn2c(=N)scc2)=O)CN(C(=O)Cn2cnnc2O)CCO1 CC1CN(C(c2cc(CO)nn2C)=O)CC1(C)C(=O)N(C1CCCC1O)C CC(C)(C#N)CC(=O)NCC1=CCN(C(=O)CC2(C(F)F)CC2)CC1 CC1CCCC(CC(=O)NCC2CC(O)(CNC(=O)CN3CCNC(=O)C3)C2)O1 N1(C(C2C(C(=O)OCC)C2)=O)CCN(C(=O)CS(C)(=O)=O)CC1C(C)C c1(C(N2CC(O)(CCNC(C3(F)CCCC3)=O)C2)=O)coc2c(F)cc(F)cc12 C1(CNC(CCOC)=O)CC2CCC1N2C(=O)C(Cc1ccccc1)N(C)C CC1CN(C(C2(C(F)F)CCOCC2)=O)CCC1NC(C1CCC(C)C1)=O C(=O)(C(F)(F)C(F)(F)F)N1CCC(NC(Cc2cccc(SCC)c2)=O)C12CC2 N1(C(CN(CC(C)C)C(c2cc(F)cnc2O)=O)=O)CC2CCOC(=O)C2C1 CC(C(=O)NC1CCCN(C(c2ccc(OC(F)F)nc2)=O)CC1)C(C)(C)C C1(NC(Cn2nnc(C)n2)=O)CCN(C(C2(C)CCN(CC(C)(C)C)C2)=O)C1C c1(OCCS(=O)(=O)N(C)C)cccc(NCCCSC(C)(C)C)c1 N1(C(CCCCC#C)=O)CCCC2C1CCN2C(C1CC(O)(c2cccs2)C1)=O CC(C)C(CC1CCCCC1)C(=O)NCC(CO)NC(c1ccc(F)cc1N)=O C1(COCCC)CCN(C(C(=O)NCC2COC2)C(C)(OC(C)(C)C)CC)CC1 c1(CCNC(=O)CC2CCN(C(=O)CCCn3ccnc3)C2)ccc(O)nc1 C1(NC(=O)CC2(O)CCOC2)Cc2cccnc2C1 C=CC1CN(C(c2cc(OCC)ccc2O)=O)CC1NC(C1COCCO1)=O C(C)(CO)(C(=O)NCC(C)(CSC)OC)NC(C(C1CCC1)OCC)=O C1(NC(COCCC(C)C)=O)CN(C(C2(C)CCCC2O)=O)CC2(CC2)C1 C1(N(C)C(C2COC2)=O)CCC(NC(C2C3COCC23)=O)CC1.C1(C(=O)N)(CF)CC1 S(=O)(=O)(c1ccc(C(=O)O)c2cnccc12)NCC(C(C)(C)C)CCS(C)(=O)=O c1(COC)ccc(C(=O)Nc2nc(C(=O)Nc3nc(C)c(Cl)s3)cs2)cc1 c1(C(N2CC3C(NC(C(C(C)C)C(C)C)=O)(C3)C2)=O)cccc2c1CCC2=O N1(CC(=O)N(C2CCCC2(F)F)C)CC(NC(c2ccc(Cl)nc2)=O)C(C)(C)C1 N1(CCOCCOCC)CCCC(NC(C2(C)CC=CCC2)=O)C1C C12(C(=O)NC3C(C)(C)CN(C(c4ccc([N+](=O)[O-])s4)=O)C3)CCCCN1CCC2 c1(C(N2C(CNC(C(C)CO)=O)CCCC2)=O)ccc2c(c1)COC(=O)N2 CC1CCCc2c(C(=O)OCCSc3ccc(F)c(F)c3)cnn21 N1(C(CC(C)OC)=O)CCC(COCCCNC(c2scnc2C)=O)CC1 c1(COC(C)(C)C)ncc(C(=O)NCC2CC(NC(C3CC3C#N)=O)C2)[nH]1 N1(C(CCOCCOCC)=O)CCC2CCN(C(=O)COCC(O)N(C)C)CC12 N1(C(C2(CC)CCCC2)=O)CCCN(C(=O)Cc2cncn2C)C(CO)C1 Cc1nc(C)n(CC(=O)NCCC2CCN(C(c3cnc(Cl)s3)=O)C2)n1 c1(CNC(C(F)(F)F)c2ccccc2)ccncc1SCc1ccccc1 c1(C(=O)NCC(C)N(C(C2N(C(C)=O)CCOC2)=O)C)cnnc2ccccc12 Cn1nccc1CC(=O)NCCC1CCC(NC(C2(CCF)CC2)=O)C1 C1(NC(c2nc(CC)oc2)=O)CC(CO)N(C(=O)C(C)C2CC2)C1 N1(C(C(C)NC(COC)=O)=O)CCC2C(CCN2C(C2(c3oncc3C)CC2)=O)C1 N1(C(C2C(C)(C)C2CO)=O)CCC(NC(=O)CC2CCCC23CC3)C(C(N)=O)C1 C1(C(=O)NC2CCCN(C(C3CC(F)C(=O)N3)=O)C2)CCc2ncnn2C1 Cc1cc[nH]c(=N)c1C(=O)NCC1CCN(C(=O)C(c2cncn2C)O)C1 CCC(F)(F)C(C)(C)C(=O)NCC12CCC(CC1)N2C(c1csc(C2CC2)n1)=O c1(C(=O)NC(C2CCN(C(c3ccc(F)cn3)=O)CC2)C)coc2c1CSC2 c1(NC(C2C=CCN2C(c2cc([N+](=O)[O-])cs2)=O)=O)cccc2nccn12 N1(C(C(CC)OC)=O)CCN(C(=O)CCCCN2CCCCC2)C(C(F)F)C1 N1(C(c2cc(C)n(C)n2)C(=O)NCc2nnn(C)n2)CCC(C)(C2CC2)C1 O=C(C1=C(c2ccccc2)CCCC1)N1CC=CC(NC(C23CCCC2C3)=O)C1 c1(OC)ccc2c(c1)C(NCc1cc(N3CCC(OC(F)F)C3)ncn1)CCO2 Cc1ccc(-c2cc(C(=O)NCC(C)NC(=O)C(=O)NCC(F)F)n[nH]2)s1 S(=O)(=O)(c1ccc(N(C)CCNC(=O)C2CC2)cc1Cl)NCC(c1cc(C)sc1)=O c1(-c2cc(C)ncc2)cn2cc(C(N3CCCC4CCCCC34)=O)ccc2n1 C1(CNC(C2N(S(C)(=O)=O)CC2)=O)CC2CCCC(C1)N2C(=O)C=CC(F)(F)F O=C1OCC2CCN(C(NC3=CCCS3)=O)C12 C1(CCCC)CN(C(c2cnc(C)n2C)=O)CCN1C(C1COCCC1(F)F)=O CCC(CC)(CC)C(=O)N1CCCN(C(c2cccc(F)c2C#N)=O)C1C n1(CC(=O)N(C(C)CNC(c2ccnn2CCF)=O)CC)cnc([N+](=O)[O-])c1 C1(CNC(C(C)CO)=O)CC2(C1)CN(C(=O)CCc1cc(Cl)cs1)C2 C(=O)(C(C1=CCC2CC2C1)NC(=O)C(c1cccc(Br)c1C)(F)F)OC CN1CC(NC(c2cn(CCNC(=O)OC(C)(C)C)cn2)=O)CC1(C)C c1(C(=O)NC2(CNC(C(C(C)C)O)=O)CCCCC2)cc2n(c1)CCOC2 C1(NC(c2n[nH]cc2Br)=O)CCCC12CCN(c1ccc(C(F)(F)F)nn1)CC2 c1(OC)ccc(OC)c(CC(=O)N(C2CC3CNC2C3)CC2(O)CCC2)c1 N1(C(CC(CC)(F)F)=O)CC(C)CN(C(=O)Cc2cccnc2Cl)C(C)C1 c1(C(=O)NCCC(C)N(C(c2n(CC)cnn2)=O)C)ccc(Br)cc1 c1(C(C)C)ncc(C(c2nnnn2C2CC2)NCc2ccno2)s1 C(C)(C)(C(C)(C)C)NC(CC1C(NC(c2cn(CC=C)nc2)=O)CCC1)=O C(=O)(CC(C)C(F)F)N1CC(N2CCN(C(=O)Nc3c(C)ocn3)CC2)C1 C1(CNC(C(C)C2CCC2)=O)CC(F)(CNC(=O)CC2CCC(O)C2)C1 CC1CN(C(c2cc(F)c[nH]2)=O)CC1CNC(=O)CCCCc1ccccc1 N1(Cc2nnc(CC)o2)CCCC(CO)(NC(=O)CCOC2CCCC2)C1 CC1=C(C(=O)NCCC2CCCN(C(C3CCCN3C3CCCC3)=O)C2)CCO1 Cc1cc(C(N2CC(NC(=O)CCCc3ccccn3)C(C)C2)=O)c(C)o1 C1(NC(C(C)CN(C)C(C2CC=CC(O)C2)=O)=O)CCOCC12CCC2 c1(C(=O)NCC2N(C(c3c(C)nc(O)[nH]3)=O)CC(O)C2)c(N)sc2ccccc12 C1(C(=O)NC2C(NC(c3n(CC)ccn3)=O)C2)CCc2nncn2CC1 C(N=c1nc2c(ncn2C)c(NC(c2nccn2C)C)[nH]1)c1cnc(C)n1C c1(C(=O)NC(C(C)NC(CCCOCC)=O)C)cc(O)c2sccc2c1 CC1CC(CNC(=O)CC23CC(C2)C3)CCN1C(=O)Cn1ccc(Br)cc1=O C12(NC(C=C(C)C3CC3)=O)CCCC1N(C(C1CNC(=O)N1)=O)CC2 N(C(=NCCOC(C)C)NCC1(C)CCCOC1)CCSC C1(C(N2CC(NC(=O)Cn3cnnc3O)C2)=O)CC2CC1CC2(F)F c1(NC2C3N(C(C(C(CC)C)C)=O)CC(CC3)C2)ncnc2scc(Br)c12 C1(CNC(C(c2cnccn2)C)=O)C2CCC(C2)N1C(c1ccc(C(N)=O)[nH]1)=O C(c1ccc(F)c(F)c1)=CC(=O)NCC(CCCC)NC(C1CCSC1)=O c1(NC(C2(NC(CC3C(C)CCC3)=O)CC(F)C2)=O)cccc(N=[N+]=[N-])c1 N1(C(CCS(C)=O)=O)CCCC(O)(CNC(=O)CN2CCCC2=O)C1 c1(C(N2C(C)CCC(NC(=O)C3=CCCSC3)C2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(OC)ccccc1C1CCN(C(C2CCCCC2C(C)(C)C)=O)CC1 CC(c1ccccc1Cl)=CC(=O)NC1CCCC(NC(=O)CC2CCNC2=O)C1 N1(C(C(COCC)C)=O)CCC2(NC(c3cnc(C)c(OC)c3)=O)CCCC12 c1(C(=O)OC)nc(Cl)[nH]c(=NCC2C(C)CCCN2C(c2cnsn2)=O)c1OC c1(C(=O)NC(CCOCC)C(=O)NCC(O)CN(C)C)c[nH]c(C#N)c1C c1(C(N2CC(C)(N(C(=O)Cc3nncn3C)C)C2)=O)cccc2oncc12 C1(C(=O)NCC(n2cc(CNC(N)=O)nn2)C)CN(C(=O)C(C)(C)C)CCO1 c1(C(C(=O)NC(CNC(CCC=CCC=C)=O)CO)(C)C)ccccc1C C(=O)(CCCc1ncco1)N(C(=O)C(c1cccs1)C1CCCO1)CC(=O)O CCC(CC)CC(F)C(=O)N1C(C(N2CCOCC(F)(F)C2)=O)CCC12CC2 Cc1ccc2sc(C(=O)NCC3(NC(C4CCCO4)=O)CCCCC3C)cc2c1 C1(CC(=O)NC2(C#C)CC2)CC2(C1)CN(C(c1csc(C)n1)=O)C2 c1(C(=O)NC(CC)(CNC(=O)C(c2cccc(Cl)c2)C)CC)cc(Cl)ncc1O c1(C(=O)NC(C)(CNC(=O)CC#N)CO)ccc2cc([N+](=O)[O-])ccc2n1 CC(CN(C(C(=O)NCc1cccs1)C1CC1c1ccccc1F)C)C(C)(C)C C=CCCCCCC(=O)N1CC=CC1CNC(=O)Cn1ncc(O)nc1=O S(=O)(=O)(c1ccc(C#N)c(N2CCCC3(CCCO3)C2)c1)NC1(C)CCOC1=O C=CCC(C(=O)N(CCCC)C)NC(C1CCC(=O)CC1)=O CC(C)CC(C)(CNC(=O)CC1CSC1)NC(c1csc(S)n1)=O C1(C(N(CC(O)CF)C)=O)CC2CC1CC2NC(C1CC2(C1)CC(O)C2)=O C(=O)(CC(CC)C(C)C)NCC(CCNC(c1cccc(CCC)c1)=O)OC C1(NC(C(C)Oc2ccc(I)cc2)=O)CCN(C)CC1c1ccnn1C c1(C(=O)Nc2cn(Cc3cccc(OC)c3)nc2C)ccc2c(C)[nH]nc2c1 N1(C(CC2(CSC)CC2)=O)C2CCC1C(C)C(NC(c1sc(C)cc1C)=O)C2 C1(NC(C2C(C)C2)=O)CCC2CN(C(=O)Cc3ccc(O)cc3)CC2C1 c1(OCC)ccccc1C(=O)NC(C)CNC(=O)COCCCOC c1(C(N(CCCC(C)C)C)=O)cnc(CNC(=O)C(F)C(C)C)nc1 N#CC1CN(C(c2cccc(O)n2)=O)CC1NC(c1cc(Cl)cnc1F)=O CCC(C(=O)OC)NC(c1nc(CNC(=O)Cc2cccnc2)cs1)=O C(C(N=[N+]=[N-])C(=O)N1CC(NC(=O)Cc2c(Cl)cccc2Cl)C(C)(C)C1)OCC CCC(C)(C(=O)NCCOC(C)(C)CNC(=O)CCC(C)OC)OC.C(=O)SCC c1(C(=O)OC)cc2ccccc2[nH]c1=NC(=O)c1cccc(C(F)(F)F)c1C c1(C(=O)NCC23CN(C(C#C)=O)C(C2)CO3)ccc(S(N)(=O)=O)o1 N1(C(c2onc(C)n2)C(=O)Nc2ccc(Cl)cc2F)CCN(C)C(C#N)C1 C1(CNC(C2(C(=O)OCC)CC2)=O)CCN(C(=O)CC2CC23CC3)C1 c1(OC)ncc(C(N2CCCN(C(c3ccnc(OC)c3F)=O)CC2)=O)cc1C c1(-n2ncc(C(N3C(CC(=O)OC)CC3)=O)n2)ccc(Cl)cc1 n1(C2(C(=O)CNC(C3C(OC(C)=O)C3)=O)CC2)cc(C2(C)COC2)nn1 O=C(C1=C2CCN=C2NC=C1)NCC1CCN(C(c2ccc(Br)cc2F)=O)C1 N1(C(c2c(C)noc2)=O)CCCCC1C1CCN(C(C2(C)CCCOC2)=O)CC1 C1(C)(CC)CC(C(N2CC=CC2CNC(=O)CC2(CSC)CC2)=O)C1 Cn1c(-c2noc(CSCCCO)n2)cc2ccc(Br)cc12 C12CS(=O)(=O)CN1C2=O.C(C)(CCCNC(C)=O)NC(C(F)=CC)=O C1(C(=O)NCC(CC)NC(=O)Cc2c(Cl)cccc2Cl)CCN(CCO)C(=O)C1 C12(NC(=O)CC(C3CC3)C3CC3)CC(CC1C(=O)O)C2 c1(CNC(CCN(CC=C)C(c2cccnc2)=O)=O)ccc(C)nc1C C1(NC(=O)CC2OCCCO2)CCCCN(C(=O)CC2CC3CC3C2)C1 C1(CNC(CCC(=O)NC2CC2)=O)CC(C(=O)N2CCC(CCO)CC2)=NO1 Cc1nc2c(cc1C(=O)N(CC(C)NC(=O)CCC(C)N(C)C)C)c(C)nn2C c1(C(N2CCC(=CCNC(C(CSC)(C)C)=O)CC2)=O)cc(Cl)c(N)cc1F C1(CC(=O)NC2CCCCC2CNC(c2ccccn2)=O)CCCNC(=O)C1 N1(C(c2nc(CCC)sc2)=O)CCC2C(C1)CN2C(C1CC(C)(C(=O)OC)C1)=O C1(NC(C2N(C(C(C3CCCC3)OC)=O)CC2C)=O)CCC(=O)NC1C C1(N(C)C(c2ccnc(O)c2)=O)CCCN(C(c2cscc2C(F)(F)F)=O)CC1 Fc1cccc(Cl)c1CCNCC1CCCC1C1CC1 C(C1(O)CCCc2ccccc21)NC(c1cccc(Br)c1Br)=O C1(C)(SCCCC)CC(NC(=O)CN(C)CCOC)CN1C(=O)C1CC1 N1(C(c2c(CC)ccs2)=O)CC2CCC1CN2C(=O)CCCCCSC N1(C(C2C(C#N)C2)=O)CCC(N)C(O)C1.c1(NC(=O)C(N)=O)cccc(S)c1 C1(NC(c2c(C)snn2)=O)CC(C)CN(C(c2cnc(O)c(Br)c2)=O)C1 c1(CC(N(C(C(=O)N(C(C)C(F)F)C)=O)C)Cc2nccs2)ccccc1 C12(NC(C=C(CCC)C)=O)CCCC1CN(C(=O)Cc1ccc(Cl)cc1)C2 N1(C(c2cc(CC)no2)=O)CCN(C(c2cnn(CC(F)(F)F)n2)=O)CCC1C O=C(N=c1[nH]oc(C2CC2)c1Br)C1(C(F)(F)F)CC2(CCC2)C1 N1(C(CC2C(C)OCC2)=O)CC=C(C(=O)NC2(C(N)=O)CCCOC2)C1 Cc1cc(C(=O)NC(C)CCNC(C2CCCCN2C)=O)cc(=O)n1C c1(C(=O)OC)coc2ccccc2c1=O.c12cccc(n1)NC21CCC1 C1(COC)(CNC(C2(C)CS(=O)(=O)C2)=O)CCN(C(c2csc(C)c2N)=O)C1 c1(C(CNC(=O)C(O)C2(N)CC2)OC)cc(Cl)cc(Br)c1 C1(NC(C2CCCC2(F)F)=O)CC2CC(C1)N(C(=O)CCOC1CC1)C2 C(CCCC(=O)NC(C)(CNC(c1ccnc(CO)c1)=O)CO)N(C(C)C)C C#CCCCCCCC(=O)NCC1C=CC(NC(=O)C(c2ccc(F)cc2)C)C1 C1(C(=O)NC2(C)CN(C(c3c(C(=O)OC)cccc3)=O)C2)CCC2(CCC2)C1 C1(C(=O)NCC(=C)F)CN(C(=O)C(C)CC2CCC2)CCO1 N1(C(=O)CCn2cc(-c3cc4ccccc4[nH]3)nn2)CCOC2(CCCSC2)C1 C1(NC(C2C(C)C2)=O)CC2CC(C1)N(C(c1csc3cncn13)=O)C2 C1(NC(c2c(CC)nc[nH]2)=O)CN(C(c2cc3cscc3s2)=O)C2CCCCC12 c1(NC(c2n(CCCC)nnn2)c2cnc[nH]2)ccc(F)c(Cl)c1 c1(OC)cc(O)c(C(N2CC(NC(=O)COC(C)(C)C)CCC2C)=O)cc1OC CC1=C(C(=O)NC2CCN(C(C3(F)CC=CC3)=O)CCC2CO)CCC(C)(C)C1 C1(NC(c2cc(C)sc2)=O)CN(C(c2cc3n(c2)CCCC3)=O)C2(CCCC2)C1 N#Cc1ccc(C(N2CCCC2CC(=O)NCCCc2nccs2)=O)o1 N1(C(C(CC)N(C)C)=O)CC(C2(NC(c3cnn(C)c3Br)=O)CC2)C1 c1(C(=O)NC2CCC(NC(C(CSC)O)=O)CC2)cc2c(F)c(F)ccc2s1 C1(NC(C(C=C)(C)C)=O)CN(C(=O)C(CC(C)C)N(C)C)CCC1O C(=O)(C(C)(O)C(C)c1ccccc1)NC1(CCNC(CSC)=O)CC1 CN1CC2CCC1CN2C(C1(N(C(C2CC3(CC3)CO2)=O)C2CC2)CCC1)=O Cc1c(C(N)=O)cccc1C(=O)NCCCC1CCCN1C(c1cc(O)cs1)=O C1(C(=O)NCc2cc(C)ns2)CC(C)(C)CCN1C(=O)C1=NNC(=O)C1 Cc1cc(O)c(C(N2CCC(CNC(=O)C3=COCCC3)C(C)C2)=O)nn1 CCCC(CC)C(C(=O)NC1CC2(C1)CC2(F)F)N(C)C(c1ccccc1)C C=CC1CN(C(=O)CC2CCN(C)CC2)CC1NC(c1ccc(NC(C)=O)s1)=O n1(CC)c(C(=O)N(CCCN(C(=O)CN2CSCCSC2)C)C)cnc1O Cc1c(C(=O)NC2CC3C(NC(c4cnn(C5CCC5)n4)=O)C3C2)cnn1C C1(CNC(CC(C)NC(N)=O)=O)C2CN(C(=O)CCCc3ccc(F)cc3)CC12 c1(CC(C)NC(N(CCOC)Cc2nccs2)=O)ccncc1 n1(CC)cc(C(N2CCC(c3cc(C)no3)C2)C(=O)NC(C)C)nn1 CC1(C)C(NC(c2cnc(S)[nH]2)=O)CC1CNC(c1cc[nH]c1C1CC1)=O C1(C(=O)NCCC(C)N2CCC2)CC2(CCN1C(c1cnnn1C)=O)CC2 N1(C(CC(=C)C)=O)CCC(F)(F)C(CNC(=O)C(C(C)C)NC(C)=O)C1 N1(CC(=O)NCC(C)CNC(=O)C(c2ccc(Cl)s2)C)CCNC1=O c1(SC)nc(C(N2CCCC2C2C(CNC(=O)C(F)C(C)C)C2)=O)c2ccccn12 CCCCCCC(=O)N1CCC(N(C)Cc2ccnc(C)n2)C1 c1(C(=O)NCC2CN(C(C(C)OCC#C)=O)CC23CCC3)cn2cnnc2cn1 C1(F)(C(N2CCC(N(C(C3CCCN(CCC)C3)=O)CC)C2)=O)CCN(C)CC1 c1(OC)ccc(Cl)c(C(=O)NC2CCCN(C(=O)C(O)P(C)(C)=O)C2)n1 C123CC4CC(C1)CC(C4)(C2)NC(=O)CN3.CC1(C)CN(C(c2cnns2)=O)C1 C1(C(=O)NCC(CC=C)NC(c2ncoc2CC)=O)CCCCN1CC(F)F C=CC(C)(CCOC)C(=O)NCC1CCCN1CCCO CS(=O)C1CN(C(c2cc([N+](=O)[O-])c(N(C)C)cc2F)=O)C2(CCC2)C1 C1(CC)CN(C(C2(O)CCOCC2)=O)CC1C(=O)N(C)CCOCC1CC1 c1(C(N2CC(CC(=O)N(C)CC3CCCC4CC34)(OC)C2)=O)ccc(O)cc1F C(=O)(C(O)CC1CCCC1)NCCCN(C(=O)CC1CCNC1=O)C c1(C(N(CCC(C(C)C)NC(CC(=C)Br)=O)C)=O)cccc2nc(C)nn12 C1(NC(c2c(C)[nH]nc2Cl)=O)CCC2CC1CN2C(c1ccnn1C(C)C)=O C1(C(N2CCCN(C(CC3(C#N)CC3)=O)CC2)=O)CCc2nnc(O)n2C1 C1(NC(c2scc(C)c2)=O)COCCN(C(=O)C(C)C(F)(F)F)C1 c1(CN2CCCC(Cc3cn(-c4cccc(C)c4)nn3)CC2)ccc(C)n(C)c1=O c1(C(N2CC(C)(C(=O)NC3CC(SC)C3)C2)=O)ncc(C)cc1C c1(C(=O)NC2(C(N3CCC(N4CC=CC4)C3)=O)CCSC2)c(F)cncc1F C12(NC(Cc3nc(C)[nH]n3)=O)CCCC1N(C(c1cc(C3CCC3)on1)=O)CC2 C(=O)(C(F)C(F)(F)F)NC(CN(C(=O)C(C(C)(C)C)n1ccnn1)C)(C)C C(CC(=O)NCC(C)(F)C(C)C)(C(C)=O)NC(C(CC=CCC)C)=O C1(C(N2CC3(CN(C(C4CC5C(C)(C)C5C4)=O)C3)C2)=O)CC2CCCCCCC12 Cc1cncn1CC(=O)NCC1CN(C(C23CC(C)C2C3)=O)C1 C1(NC(CN(C)C(N)=O)=O)CC(NC(=O)CCCCC2CC2)CC1O C1(NC(c2ncc(C)cc2C)=O)CCC(O)CN(C(c2scnc2C2CC2)=O)C1 N1(C(C(C)NC(CC)=O)=O)CCCCC12CC(NC(c1ccc(Cl)c(N)c1)=O)C2 C(C1c2ccccc2CN1C(=O)C1=CCOCC1)NC(C(CC=C)C(C)C)=O C1(C(=O)NC)CCCC12CC2.n1(C(C)C)nnnc1-c1ccccc1.N12CCC1C2 C1(NC(C2C(C)(COC)C2)=O)CCCC12CN(C(=O)CCn1ccnc1)C2 N1(C(C)=O)CCCC(C(=O)NC2CCC(NC(C3CCCN3C)=O)CC2)C1 CCCCC(C)C(=O)N1CC(NC(=O)C(F)C(C)(F)F)CCC1C c1(CNC(C2C(CNC(CCCOC)=O)CCC2)=O)cnn(C)c1C c1(N(C(C)(C)C)C(N2C(CCC(C)N(C)C)CC2)=O)cccc(C#N)c1 C1(CNC(C2C(C(C)(F)F)C2)=O)CC(NC(=O)CCCC2CCOCC2)CC1O C#CC1(C(=O)N(C2CC(NC(c3cc(C(C)C)oc3C(C)C)=O)C2)C)CCCC1 C1(NC(CCCOC(C)C)=O)CN(C(c2ccnn2C(C)C)=O)CC1C C1(C(=O)NC(CNC(C=COCC)=O)CCOC)(OC)CC(C)(C)C1 CC(C)C(CC(=O)NCC1CCCCO1)NC(=O)C(C)C1(O)CCC1 C1(C(=O)NC(c2ccc(CNC(c3ccncn3)=O)cc2)C)CCC(F)(F)CC1 C1(CC(=O)NCc2cncc(C(N3C(C(=O)NC)C=CC3)=O)c2)NC(=O)NC1=O C(C(C)(C)CNC(=O)CC1CCCC1C)N(C(=O)CNc1ncccn1)CC N1(C(C2C(OCC)C2)=O)CC2(CCCC(CNC(c3ncc(Cl)n3C)=O)O2)C1 c1(C(=O)OC)cnc(S(=O)(=O)Cc2cnn(C3CCCC3)c2)s1 C(=O)(CS(=O)(=O)C1CCCC1)NCC1(C)CCCN1C(C1CC2CC1C2)=O c1(C(N)=O)cccc(COC(=O)CC(O)c2cnc(Cl)s2)c1 N1(C(CNC(=O)OCC=C)=O)CCCC(O)(CNC(C2CN(C(C)=O)C2)=O)C1 C1(C(N2C(c3ncc[nH]3)CC(OC)C2)=O)CCCNS1(=O)=O CC(C)C(C(=O)N1CCC1(C)CCO)NC(=O)Cc1cn(C)nn1 C1(C)(CNC(CCCOCC)=O)CN(c2ccc(C(=O)OC)c(C)n2)CCO1 N1(C(C(C=C)C)=O)CCN(C(=O)Cc2cccc(C)c2)C(C)C1C N1(C(C2(COC)CCCO2)=O)CCC(F)(F)C(CNC(=O)CCCC2CC2)C1 c1(C(C)C)cccc(C(F)(F)F)c1.c12noc(n1)CC1(CCOC1)NC2 Cc1cc(C(N2CCC(C)(NC(=O)C(F)F)CC2)=O)cnc1C(F)(F)F C(=O)(CCC(CC)CC)NCC(C)(C1CCC1)NC(c1c(CCCC)ocn1)=O C1(CC(=O)NCc2nc[nH]n2)(NC(C(COC(C)=O)C)=O)CCCCC1 c1(C(=O)NCC2(CNC(C=Cc3nnn(C)n3)=O)CCC2)cccc2oc(=N)[nH]c12 N1(C(CC2N(C(CCC3CC(OC)C3)=O)CCCC2)=O)C2C=CCC1CC2 C1(C(=O)NC(COCC)C(=O)NC(C)C(C)(C)CO)CC2C=CC1C2 C#CCCC(C(=O)OC)NC(C1CC(O)CN1C(=O)CC1C=CCCC1)=O C=CC1OCCC1C(N1CCOCC1CC(=O)NC(c1ccnn1C)C)=O c1(CCCC)ocnc1C(N1CC(CCNC(=O)CC(C)C2CC2)C1)=O N1(C(C2(CC)CCCCC2)=O)CC2CCCC(CNC(=O)Cn3nccn3)C2C1 c1(C(N2C(CNC(C(CC(=O)OC)C)=O)CCC2)=O)cccc(C)c1NC C(=O)(C1=C(c2cnn(C)c2)N(CCF)C(=O)NC1c1cccc(=S)n1O)OCC c1(C(N(C)CC2N(C(c3cc(CCC)on3)=O)CCC2)=O)cccc(Cl)c1O N1(C(c2c(CC)noc2)=O)CC2CCC2(NC(=O)C(C)=C2CC2)C1 C1(NC(CCCCOCC)=O)CCN(C(=O)CC2CCCC2O)CC1CO C12(CNC(C=C3CCC(C)C3)=O)CN(C(=O)C=Cc3ccccn3)CC1CCO2 N1(C(c2cccc(F)c2Br)=O)CCC2C1CCCN2C(c1c(O)cccc1O)=O N1(C(CC(COC)C)=O)CCC(CCNC(=O)C(C)=C(C)C)C(F)(F)CC1 C1(CNC(=O)NC2CC(C#N)C2)CCN(Cc2ccccc2)C1c1ccccc1 C=CCC(CC(C)C)C(=O)N1CCN(C(=O)CSCC(=O)NCCC)CC1CO C12(C(=O)NC(C(=O)NCc3cc(C(C)C)on3)CC3CCC3)CC1CNC2=O c1(CNC(C(C2CC2)NC(c2c(C)csc2)=O)=O)ncc(F)cn1 CCC(CC(F)F)C(=O)NC(C1CCCC1)CNC(=O)C=Cc1cocn1 C1(NC(c2cc[n+]([O-])cc2)=O)CC1C1CCN(C(c2cc3n(n2)CCC3)=O)CC1 Cn1cc(C=CC(=O)NCC(C2CC2)NC(=O)CSCc2cccc(F)c2)cn1 c1(CN=C(NC(C)(C)C)NC2CC2C2CCC(=O)NC2)ccnc(O)c1 n1(CC#C)c(N(CCOC)CC)nnc1CS(N)(=O)=O CON1CCC(NC(=O)C(C(C)CC)N(C)C(c2cc(=O)cc[nH]2)=O)CC1 C1(OCC(=O)N(CCC)C2CC2)CN(C(=O)C=CCN2CCCC2)C1 CCCCCC(=O)NCCOCC(N1CCC(OC2(C#N)CC2(C)C)CC1)=O C=C(C)CCC(=O)NCC1CCN1C(c1c(C)coc1C(C)C)=O C1(CNC(CC=CCC)=O)CN(C(C2(CO)CCOCC2)=O)CCCO1 C=CC1COCC1NC(=O)CN(C(C1COCCC1C)=O)C(C)C C(=O)(C1=C(CCOC)N(C(C2CC2)C)C(=S)NC1c1cscn1)OCC c1(SC)ccccc1NC(N1CCC(CN(C)C(c2ccncc2F)=O)CC1)=O c1(CC)oc(C(=O)NC2CCCC2CNC(=O)CCc2ccc(C)o2)cc1C CC12CCCC1NC2.c1(C(=O)NCC2CC(F)(F)CO2)ccccc1Cl CC(C)(C)C(O)CNC(C1(NC(=O)C=CC(F)F)CSC1)=O C(=O)(C(C(C)(C)O)NC(C1CC2(CCC2O)C1)=O)N1CC(C#C)(C(N)=O)C1 C(=O)(CCCCC(C)(C)C)N(C1CCC2CN(C(=O)C(F)OC(F)(F)F)CC12)C c1(C(C)NC(C2CCN2Cc2ncco2)=O)ccc(F)cc1 c1(C(N2CCC(=C)CC2C(=O)NC2(CSC)CC2)=O)cc2ccccc2[nH]1 O=C(CCS(=O)(=O)C(F)(F)F)NC1CC(NC(C2CC23CCS(=O)(=O)CC3)=O)C1 C1(C)(CNC(C(CC)F)=O)CCN(C(=O)CC2CCCC(=O)N2)CC1 CC1C(N=c2[nH]c(=NCC3(N4CCCCC4=O)CC3)[nH]c3c2COC3)CCN1C c1(-c2ncc(C(N3CC(O)(C(C)NC(C=CCOC)=O)C3)=O)s2)ccccc1C C#CCC(CC#C)C(=O)N1CCCC(NC(=O)C(c2ccc(Cl)cc2)(C)O)C1 C1(C(=O)NC2CC(CCNC(C=C(C)C)=O)C2)(Cc2snnc2C)CCOCC1 C1(C(=O)NCC2CN(C(C(C)CN(C)C)=O)CC2O)CCC([N+](=O)[O-])CC1 c1(SCC(N2CC(O)(CNC(=O)CC(O)C3CC3)C2)=O)ccc(F)cc1 O=S(=O)(c1nc(N2CCCC(CO)C2)ccc1Br)NCCC(O)C1CCCC1 Cc1ccc(O)cc1NC(C1COCCN1C(=O)CSc1ccccc1)=O C1(NC(C(C)=C(CC)C)=O)CC2CC(NC(c3c(N)ccc(F)c3C)=O)CC2C1 N1(C(C=CC=CC)=O)CCC(O)(CN(C)C(C2COCCC2C)=O)CC1 CCC(C)CC(C)C(=O)N(C1CCC2CN(C(C3CC(C)CC(C)C3)=O)CC12)C c1(C(=O)NC(C)C(C)NC(C2CCOC2)=O)ccc(Br)c([N+](=O)[O-])c1 C1(CC(=O)N(CC(CNC(C2(CC#C)CCCC2)=O)C)C)CCCC(C2CC2)O1 c1(CNC(c2cc(C)[nH]n2)=O)nc(CNC(=O)CCN2CCC(F)C2)cc(O)n1 C1(C(=O)NC2(CCC(=O)NCCC34CC(CO3)C4)CCC2)CCCC1C(F)F C(=O)(C(C)(F)C(C)(C)F)NC1CN(C(CC(C)O)=O)CC1F Cc1nc(C=CC(=O)NC2CN(C(C3CCCC(C)(C)C3)=O)CC23CC3)[nH]c1C N1(C(CC(CC)O)=O)CCc2cccc(-c3cn(CC4CCOC4)nn3)c21 c1(OC)ccc(C(=O)NCC2CCN(Cc3cnc(Cl)s3)C2)c(OC)c1 C12(COC)CC(CNC(=O)C(C)(C)C)(CN1C(=O)CC1CCC(=O)CC1)C2 c1(C(=O)NC2(C)CC(NC(C(C)OCC(C)C)=O)C2)cc2ccncc2c(O)n1 c1(NC(C2N(C(C(C)Cc3ccco3)=O)CCC(O)C2)=O)ccc(Cl)c(C#N)n1 N1(C(C(C=CC)O)=O)CC2CCC1(CNC(=O)CC(C)OC)CC2 c1(C(=O)NC(CCNC(C(C)OCC)=O)C)ccc2c(c1)COCO2 N1(C(CC)=O)CCC(C(=O)N(CC(C2CC2)OC)CC)CC1 N1(C(Cc2nc(C(C)(C)C)sc2)=O)CCC2CCC12CNC(=O)C(C)(C)C1CC1 c1(CC)cn2c(n1)CC(C(=O)NCCN(C(=O)Cn1cnnn1)C(C)C)CC2 n1(CC=C)nc(-c2ccc(Br)cn2)nc1C(c1cncnc1)C c1(N2CCN(C3C(C=C)OCC3)CC2)cccc(S(=O)(=O)N2CCC(SC)C2)n1 N1(C(c2cc(CC)sn2)=O)CCOCC1CNC(c1cccc(C)c1)=O N1(C(C(C)OC)=O)CCC2(CC1)CC(CN(C)C(c1ccc(CO)o1)=O)C2 c1(N(CC)CC)ccc(C(=O)NCC2CCNC(C)C2)c(O)c1 C1(CC)CN(C(c2cnc(N)c(CO)c2)=O)CCN1C(C1CCC(=O)NC1)=O c1(NC(C2CCN(C(CCCC#C)=O)C2(C)C)=O)cn(C)c(=O)cc1C c1(C(=O)NC)cc(NCC2CCCN2C(=O)CCC2(C)CC2)ccc1F c1(C(N(C2CCCCC2)CCNC(C(C)N(C(C)=O)C)=O)=O)occ2c1CCC2 c1(CC)cnccc1C(=O)NCC=CCNC(c1cn(CC(F)(F)F)nc1C)=O c1(C(=O)NC(C)CCNC(C2(CF)CC2)=O)cc(-c2cnn(C)c2)on1 C1(C(C)NC(=O)NC2CN(C(C)C)C2)CCN(c2ccc(Br)cn2)CC1 c1(C(=O)NC(C(=O)NCCCN(CC)CC)CC2CC2)cn(C)cc1C N#Cc1ccc(CNC2CC(C(=O)O)C2(C)C)c(Br)c1 CC(C)C(C(C)NC(C1C2(CC2)C12CC2)=O)NC(=O)Cn1ncccc1=O Cc1cc(C(F)(F)F)ccc1-c1csc(C(=O)Nc2cc(F)c(Cl)cn2)c1 c12cc(nc(OC)n1)NC(=O)c1ccn(n1)C1CCC(C1)NC2=O.COCO N1(C(C(CSC)C)=O)CCN(C(=O)CN2CCCC2)CC1c1cc(F)ccc1F c1(C(=O)NC2CCN(C(C(c3ccc(C)cc3)C)=O)CC2)ccc(C)cc1C Cc1nnc2sc(COC(C3CCCN(CC(=O)NCC(C)C)C3)=O)nn2c1=O Cc1ccc2c(c1)C(C(=O)NC1CC(NC(c3cnc(C(C)C)s3)=O)C1)C2 N1(C(C2CCC(CC)O2)=O)CCC2(CC2NC(c2cc(C)n(C)n2)=O)C1 N1(Cc2n(C)ccn2)CCOCC1C(=O)Nc1cncc(F)c1 CCC(C(=O)N1CCC(O)(CNC(c2nccc3[nH]ccc23)=O)C1)C(C)(C)CC C1(CNC(C(C2CC2)OCC)=O)COCCN(C(c2cc(Br)cn2C)=O)C1 CC1(C)CCCC(C)(CN2CC(C(=O)N(C)C)C(O)C2)C1 N1(C(c2cc(C(N)=O)oc2)=O)CC2(CCCC2NC(c2cc(Cl)sc2Cl)=O)C1 n1(CCN(CC)CC)nccc1C(=O)NC(C)CS(C)=O.C1C(=O)N1 CC12CN(C(=O)C=CBr)CC1(C)CN(C(C1CC3(CC3)C1)=O)C2 c1(C(N(C(C)CNC(C2CCS(=O)(=O)C2)=O)CC)=O)ccc(C(C)C)cn1 C12(C(=O)Nc3c(CC)cccc3)CCOC1CN(C(=O)N(C)CC1CCCN1)C2 CCCCCCC(CC)NC(=O)C(O)CNC(=O)C(C)(C)C(N)=O CC1CCC(NC(c2ncsc2C(F)(F)F)=O)CN1C(C1CC1C1CC1C)=O C1(C(N(CC(CNC(CC(C)SC)=O)O)C)=O)C2(CCC2)C12CCC2 C1(C(N(C)C)=O)COCCN1C(C1C2CC=CCC12)C(=O)NCC(F)F Cc1cc(C)n(C)c(=O)c1CNC(=O)NCC(O)CC(F)(F)F c1(CC)cc(C(=O)NC2(CC(N3CCC(F)(CF)C3)=O)CC2)nn1C Cc1ccc(-n2nc(-c3cnn(C)c3)nc2C2CCN(CC(F)(F)F)C2)cc1C c1(-c2cn(C3CN(C(c4nc(COC)[nH]n4)=O)C3)nn2)cnc(SC)nc1 c1(CC)ccc(C=CC(N2CC(O)(CNC(c3cc(CC(C)C)on3)=O)C2)=O)o1 CCCC(CCCNC(=O)C=Cc1csc(C(F)F)c1)NC(=O)C(C)S(C)(=O)=O N1(C(C2(CC(C)=O)CC2)=O)CC(CNC(=O)C=Cc2ccccc2F)OC(C)C1 C(C(CCN=c1nc2c(ncn2C)c(NCc2nc(C(N)=O)co2)[nH]1)OC)OC CCCCC(CC)C(=O)N1CCCOC(CNC(C2CCC2)=O)C1 CCCCC(CCCC)C(=O)NC1CC2CN(C(c3cccc(Cl)c3)=O)CC12 Cc1ccc2c(c1)C(Nc1nc3c(Br)cccc3s1)CC2 Cc1[nH]c(C(=O)NC(C)CNC(=O)C(c2ccc(F)cc2)(C)O)c(C)c1C C(C(=O)N1CCC(C(F)F)(CNC(c2occc2F)=O)C1)(C(C)C)SCC c1(CC(=O)N(CCNC(C(n2c(C)ccn2)C)=O)C2CC2)ccc2nsnc2c1 C1C(F)(F)C(=O)O1.C#CC1(OCC)COC1.C1C(=O)O1 Cc1nc(C)c(CNC(=O)NCC2(C)CSC2)[nH]1 C=CCC(C(=O)N1CCCCCC1)NC(c1cc(OC)cs1)=O C1(OC)CC2CCC(C1)N2C(C12CC1CN(C(=O)CCCn1ccnc1)C2)=O N(C(=NCCc1ccccn1)NCCF)CC(CO)Cc1ccccc1 c1(C(N2CC(NC(C34CC=CC(C3)OC4)=O)C2)=O)noc2cc(Cl)ccc12 C1(CNC(c2nn(CC)c(O)c2)=O)CN(C(c2cn(C)cn2)=O)CC(C)(C)O1 C(N=c1[nH]c(=NC(C)C(CC)CC)[nH]c2c1CC(C)CC2)c1c(CC)con1 Cc1nn(C)c2sc(C(=O)NCC3CN(C(c4nc(Br)c[nH]4)=O)CCO3)cc12 c1(C(=O)NCC(CC(=O)NC(C(CC)CC)C)O)nccc2[nH]ccc12 c1(CCC(N2CC(C)(N(C(CCC(C)C)=O)C3CC3)C2)=O)ccc2c(c1)CCO2 C1(N(CCN(CCN(C)C(=O)NCC)O)C2CC2)CC1(C)C N1(C(=O)OC(C)(C)C)CCC2(CC1)CNCCCN2C(=O)C1=CCCC1 c1(C(C(=O)NCC(C)(C)NC(c2ccc(SC)o2)=O)OC)ccc(Cl)cc1Cl C1(F)(CNC(C(CO)OC)=O)CCC(NC(=O)CNC=O)C1 C12(CNC(C(CCC)O)=O)CCC(CC1)CN2C(c1cc(N)c(F)cc1F)=O C1(CC(=O)NC(CNC(C(C)N(C(C)=O)C)=O)(C)CO)CCC2CC1C2(C)C N1(C(C2CCCCC(=O)N2)=O)CC2CCN(C(=O)C(c3cccnc3)O)CC2C1 c1(C(N2CCC(NC(c3cc(C)n(C)n3)=O)C(O)C2)=O)n[nH]c2c1CCSC2 c1(NC(c2ccc(CNC(=O)CCc3ccsc3)s2)=O)cccc(Cl)c1 C(=O)(C(O)CCC(F)(F)F)NCCCCC1CN(C)C1.c1(CC)cnoc1C(=O)N CCC1(CC)CN1.C1(CNC(=O)OC(C)(C)C)CCN(C(C)=O)C1C CCC(CC)(CC)C(c1nnnn1C(C)(C)C)NC(c1ccc(F)cc1)C1CC1 Cc1ccc(C(=O)Nc2ccc(-c3ccccc3C#N)nc2)cc1F C=Cc1cnn(C)c1C(=O)NC1CCCCC1CNC(c1coc(N(C)C)n1)=O C=C(C)C(CC(=O)NC)OC.C1(C(c2ncccn2)O)CCN(C)CC1 n1(CC)nc(C(N2CCCC(C(=O)NC(C)(COC)CCO)C2)=O)cc1O c1(CNC(C(n2cc(CC3CCCCN3C)nn2)C)=O)cccc(C(C)(C)C)n1 C(CCCCC(=O)NCCC(C)NC(c1nccnc1CC)=O)OCC C1(C(=O)NC2CC(C(=O)NCC(O)(C3CC3)C3CC3)C2)CCOCC1 c1(C(N2CC3N(C(CC(CC)C)=O)CC(C3)C2)=O)ccc(S(=O)(=O)N(C)C)cc1 C1(NC(C(c2ccc(C)o2)C)=O)CCC(NC(c2cc(C(C)C)nn2C)=O)CC1 C#CCC(CC#C)C(=O)N1CCCC(N(CCO)C(c2c[nH]c(C(N)=O)c2)=O)C1 c1(C(=O)OC)cc(CN2CC(O)CC2C(=O)Nc2cc(F)ccc2Cl)ccc1Cl N1(Cc2cccc(SC)c2)CCC2(CC1)CC(N(C)CCO)C2 Cn1ncc(C(=O)NCC2CN(C(=O)CN3C(=O)CCC3=O)C2)c1C1CC1 N1(C(CC(C)=C(C)C)=O)CCC(C(=O)NCc2nnc(O)o2)CC1C1CC1 c1(NCC2CC(=O)N(CC)C2c2cccc(C)c2C)ccc2c(cnn2C(F)F)c1 CC1CC(NC(c2cccc(Cl)n2)=O)CN1C(=O)C(C1CCCCC1)O C1(CNC(c2cc(-c3ccoc3)on2)=O)CCC2(CCC2)C1NC(=O)C1=CCC1 O=C(CC1NC(=O)c2ccccc21)NCCN(C(=O)CC1CC2(CC2)C1)C1CC1 c1ccc(CCF)cc1.C1(C(=O)NC2CC2)(CC)CN(C(C2CCC2OCC)=O)C1 c1(SCC)cccnc1C(=O)NCC1C(C)CCN1C(=O)C(F)OC c1(CNC(CCC2(NC(C(C)CN(C)C)=O)CCC2)=O)cc(O)ncn1 C1(NC(C(C)OCC=C)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC1C(F)(F)F C(=O)(C(C(C)(F)F)c1ccccc1)N(CCOCC)CCNC(=O)C(=O)N(C)C c1(CNC(C(C)OCCOC)=O)cc[nH]c1C(=O)NC(C)CC(=O)OC C1(NC(CC2CC(NC(CCn3ccc(C)c3)=O)C2)=O)CC2C(O)C(O)CC12 c1(C(C)(C)C)ccc(C(=O)NC2COCC2CNC(C2CCC2)=O)s1 C1(C(=O)NCC2CC2Cl)CN(C(C23CC2CNC3=O)=O)CC12CCC2 N1(C(C2N(S(C)(=O)=O)CCC2)=O)CCN(C(=O)C#CC2(CO)CC2)CC1C(F)F N1(CC)CCOC(C(=O)NC2(C)CC(NC(=O)CC3COCCO3)C2)C1 Cc1ccc(C)c2[nH]c(C(=O)NCCN(C(C3CC3c3ccco3)=O)C3CC3)cc12 N1(C(=O)C=CCN2CCOCC2)CCC2CN(C(C3C(F)(F)C34CC4)=O)CC2C1 C(=O)(C1CCc2ccccc21)NC1C(NC(C2CC(=O)Nc3c2cccc3)=O)C1 c1(CC)cc(C(=O)NC2CCCCC2NC(=O)C=C(C)Cl)nn1-c1ccccc1 CC1CCCCN1CC(=O)NCC1(O)CCN(C(=O)CCNC(N)=O)C1 C1(C(C)NC(=O)CC2CC2(C)C)CCCCN1C(=O)CCc1cnco1 C1(C(=O)OCC)CCN(C(C2CC(O)(CO)C2)=O)CC1 C(=O)(CC1=CSC2=NCCN12)NCC(C(C)C)NC(c1cccc(=O)n1O)=O N1(C(C2(C(C)=O)CC2)=O)CCC(C)(Cc2cn(CCC3CCCC3(F)F)nn2)C1 N1(C(C(C2CCOC2)OCC)=O)CC(n2cc(OC)nn2)C(CC)C1.C12(CC1)CO2 C(CCCCC(=O)OC1C(=O)CC1C(C)C)c1cccc(OC)c1 N1(C(C(CCCC)NC(C)=O)=O)CCC2CN(C(=O)CC(CCC)CCC)CC2C1 C1(C(=O)NCc2cc(C)[nH]n2)CCOCCN1C(=O)COCCC(C)C c1(C(N2CCCC(N(C(C=CCOC)=O)CCF)C2)=O)ccnc(Cl)c1N C#CCCCC(C)C(=O)N(C)CCOCCC(=O)NCc1ccc(C#N)o1 c1(OCCCC)ccc(C(=O)NC2CC2NC(c2scnc2Cl)=O)cc1Cl c1(SCC(=O)NC2(CNC(C(C)n3cccc3)=O)CCOC2)ccccc1O C(C(C)(C(C)C)NC(c1cn(C2CC2)nn1)=O)NC(c1c(C(C)C)snn1)=O c1(NC(=O)NCc2c(C)nc(C3CC3)nc2C)ccnc2ncc(Br)cc12 c1(CCCC)nc(C(=O)NCC2(NC(c3ccc(CO)o3)=O)CC2)cs1 CC(C(=O)N1CC(NC(=O)CN(C)C(N)=O)C(CC(C)(C)C)C1)C(C)(C)C C12(C(N(C3CCCC3)CC=C)=O)CC(CN1C(C1C3CCCC13)=O)C2 C1(NC(C(CC)O)=O)CN(C(c2cc(C)c[nH]2)=O)CC1n1ccnn1 c1(OC)ccnc(-c2cccc(C(=O)NC(C)C3CC3)c2)n1 N1(C(CC(CC)CN(C)C)=O)CCCC(N=c2cc(C)[nH]c(C(F)(F)F)n2)(CO)C1 c1(C(N2CCC(C)C(NC(=O)C(C)(C)F)C2C)=O)c(F)cccc1[N+](=O)[O-] n1(CC(=O)NCCCNC(C2CCCC2O)=O)nnc(C2CC2)n1.c1(S)ccccc1 CCCN=c1[nH]c2c(cnn2C)n1CC(=O)NC1(C2CCC(=O)NC2)CC1 C=CCC(C(=O)NCC1CC1CC(=O)N(C1CS(=O)(=O)C1)C)C(C)C C(=O)(C1=C(F)CN(C(=O)CC(O)CC(C)(C)C)CC1)N1CC(NC(C)=O)C1 C(=O)(C(CCC1CCC1)NC(C1CN(C)CCO1)=O)NC(c1c(C)ncs1)C C(=O)(C1CCCc2nncn21)N(CCN(C(C(CC=C)C)=O)C)C C12CCN(CC1)CC(=O)N2.n1(CC(C2CCOC2)OC)cc(C2CCOC2)nn1 N(C(=NCCF)NC1CCOC1C)C(CC)CC N1(C(Cc2c(C)ocn2)=O)CC2CN(C(=O)C=Cc3ccc(Br)cc3Cl)CC2C1 C=C1CC2(C1)C(=O)NC2.N1(C(c2cc(OCCO)no2)=O)CC2CC2C1 c1(C(C)OCC)nc(C(Cc2cnn(C)c2)OC)n(-c2cnnn2C)n1 CCCCCC(O)C(C)C(=O)NCCC1CCN(C(=O)CCC2CCCC2)C1 c1(C(=O)NCC(C2CC2)NC(C2CC(CC)(CC)C2)=O)cnn(C)c1C(F)(F)F c1(CCC)ccc(CC(N2CC(NC(C3(CC(C)C)CC3)=O)C(SC)C2)=O)cc1 Cc1ccc(NC(C2(NC(=O)Cc3ocnc3C3CC3)CCCC2C)=O)cc1F c1(C(N)=O)coc(CNC(=O)C(C)(C)NC(C2CCCCO2)=O)c1 CCC(C)(C(=O)N1CC=C(CNC(c2coc(=O)[nH]2)=O)CC1)C(N)=O c1(Nc2nc(C3N(C(Cc4cc(C)on4)=O)CCC3)sc2)nccnc1O c1(C(=O)NCC2C(C)CN(C(=O)CC3CCC(C)C3)C2)ccc(P(C)(C)=O)o1 C(N=c1[nH]c(=NC2CCC(=O)NC2)[nH]c2c1COC2)C1COCC(C)(C)O1 C1(OCCNC(=O)OC)CCN(C(=O)CNC(=O)NC2CC2)CC1 C1(C(=O)NC(C2CN(C(c3cccnc3F)=O)C2)C)CNC(=O)N1C CCC(CC(F)(F)F)C(=O)N1CC(NC(c2c[nH]c(Br)c2)=O)C(N=[N+]=[N-])C1 c1(C(N2CCCCC(N(C(=O)CCS(C)=O)C)C2)=O)cnc2c(F)cccn12 c1(CC(C)NC(C)=O)ccc2c(c1)OCO2.C1(c2cccs2)CC(=O)N1 C(=O)(C(C)(C)CC(F)F)NC1CCC(NC(C2(CC)CCNC2=O)=O)CC1 N(C(=NCC1(C)CCCCO1)NC1CCN(C(N2CC=CC2)=O)CC1)C(C)C C1(C(N(C(C2CCCC2)C)C)=O)CCC(C2CC2)N1C(C1CC=CC1)=O c1(NC(CC2CN(Cc3cncc(NC)c3)C2)=O)cccc(OC)c1C c1(OC(C)C(=O)N(C)CCN(C(=O)CN2CCC(C)CC2)C)cccc(Br)c1 C1(OCC(CC)(C)O)CCC2(CC2)N1C(=O)CCCON=C(C)COC Cc1ccc(N)c(C(N2CCC(NC(=O)C(C)Oc3cccnc3)C2)=O)c1F c1(NCC2N(C(c3ccc(OC)c(F)c3)=O)CC(O)C2)nc(C)ccc1C#N CC1(C)CCC(C(N2CC(O)CC2CNC(c2nccc(Cl)c2O)=O)=O)CC1 c1(C(N(C(CCNC(C(CC)(C)OC)=O)C)C)=O)cccc(F)c1C(F)(F)F C1(CCNC2(c3nnnn3C)C(CCC)CC2)CCS(=O)(=O)CC1 C1(C(N2C(CNC(C3(C#C)CCC3)=O)COCC2)=O)CNC(=O)CC1(C)C c1(C(=O)OC(C)(C)C)cc(NC(c2cn(CC3CCOC3)nn2)=O)c(Br)cn1 c1(C(N2C(C)C(NC(=O)OC(C)(C)C)CC2)=O)ccc(S(N)(=O)=O)cc1 c1(SC)cccc(CN(C(c2ccnn2C)C(N2CCCCC2)=O)C)c1 CC1CC(C(=O)NCC(N2CCC2(C)CC(=O)NC2CCC2)=O)CCS1 c1(NC(CC2(C)CN(Cc3c(Cl)cncc3Cl)C2)=O)cc(F)ccc1Br N1(CC2OCCN(CC)C2)CCC2(CC1)CC2C(=O)NC1(C)CCS(=O)(=O)C1 N1(C(c2cnc(-c3cccs3)o2)=O)CCN(C(=O)CSC2CCC2)C(CC2CC2)C1 c1(C(=O)NCC2C=CCN2C(C2CC2c2ccccc2)=O)cc2scnc2[nH]1 c1(CC(C(=O)OC)NCCS(CC)=O)c[nH]c2cc(F)ccc12 C1(CNC(CSC(C)C)=O)CN(C(=O)CSCc2cccnc2)C2(CCC2)C1 CN1CCC(C)(C(=O)NCCCNC(C2(C)CC3CC3C2)=O)C1 O=C1CN(CC2CCCN2C2CC2)c2ccccc2N1C(=O)c1cccc(I)c1 Cn1nc2c(c1N)CN(C(=O)NC1C3Cc4ccccc4C13)C2 C1(NC(c2ccc(C)cc2)=O)CN(C(c2ccc(C)cc2)=O)CC12CCOCC2 c1(NC(=O)NC2CC2c2nc3ccccc3[nH]2)nccc2occc12 N1(C(C2CCCC(C)(C)O2)=O)Cc2ccnn2CC(NC(=O)CNC=O)C1 c1(OC)ccnc(C(=O)NC2CC(CCNC(=O)COCCCF)C2)n1 CC(C)C(C)C(C)CC(=O)N1CC2CC1C2NC(c1ccc2occc2c1)=O c1(CC(N2C3CC(NC(C=NOC)=O)CC2CC3)=O)cnc2n1CCCC2C Cc1ccccc1C=CC(N1CC(N(C)C(c2cc(C(C)C)ccc2F)=O)C1)=O N1(CCC)CC(C(N2CC(CNC(=O)C(=Cc3cscn3)F)(OC)C2)=O)CC1=O C1(CNC(CC2CC(NS(C)(=O)=O)C2)=O)CCN(C(=O)CCC(N)=O)CC1 c1(C(=O)NC(C(C)NC(=O)CC2CCCCC23CC3)CO)cc(C#N)ccc1N O=S(=O)(c1c[nH]ccc1=NC1CC2(CCC2)C1)N1CCCC(C2(O)CCC2)C1 Cc1noc(CCC(=O)NCCC2(NC(c3cc(C(C)C)[nH]n3)=O)CC2)n1 C#CCCCCC(=O)N1CC=C(C(=O)NC(CO)CC=C)C1 C(CCC1CCC1)(C(=O)N(C)CCC1CCCO1)NC(C(CO)OC)=O n1(C(C(=O)OC)C)nc(CC(C)(C)C)nc1-c1cncnc1C N1(C(CCC)=O)CCC(C(=O)NCC(C)(C)NC(=O)C(C)(C)SCC(C)C)CC1 N1(CC)CCCC1C1CCCN1C(=O)Cn1nnc(C(=O)NC)c1C n1(CC(=O)OCC)cc(C2(C(=O)NC3CCCC3F)CC2)nn1.C(C)(C)(C)OC(=O)N C12(C(=O)NCC(c3cccc(Cl)c3)NC(CC(C)C3CC3)=O)CC(CCO1)C2 C1(C(N(C(C(=O)NCC(C)F)=O)C)C)CCNCC1 CCC(CCC(=O)NCC(c1ccccc1OC)NC(=O)CCn1cnnn1)OC C(CC(C)N=c1nc(N(C)Cc2ncc(Cl)n2C)c2c([nH]1)CCCC2)N(C)CC S(=O)(=O)(c1ccc(N2CCC(OC)CC2)c(C#N)c1)NCC(C(CC)C)O N1(c2ccccn2)CCC2(CCCN2CCc2cn[nH]c2)CC1 C(=O)(C1=CCOCC1)N(C1CN(C(=O)C(c2cscn2)N(C)C)C1)C CC(C)CC(C)NC(=O)CN(C)C.C(C)(C)(C)OC(=O)NC c1(NC(C2C(NCc3cccc(C(C)(C)O)c3)C2)=O)ccc(Cl)c(C#N)n1 c1(C(=O)NCCCN(C)C(c2cnc(O)o2)=O)cc2c(cn1)NC(=O)CO2 C=CC1OCCCC1C(=O)NC1(c2ccccc2)CC(NC(=O)CN2CC=CC2)C1 c1(C2CN2)cccc2c1OCCO2.N1(C(=O)OC(C)(C)C)CCN(CCF)CC1 Cc1coc(C(=O)NCC2(NC(C34CCCC3C4)=O)CCOC2)c1C Cc1ccc(Cl)c(OCC(=O)NCC2CCN2C(c2cccc(O)n2)=O)c1 C(=O)(C1=C(F)CN(C(C2(C)CC2(F)F)=O)CC1)NCc1n(CC)nnn1 Cc1nn(C)c(C)c1C(=O)C(=O)NCC1(NC(C2CC2c2nc[nH]n2)=O)CCC1 Cc1c(C(C)NC(=O)CCCn2cc(C3(O)CCOC3)nn2)cccc1F C1(CNC(c2cncc(C)c2)=O)CCN(C(c2nnn(C)n2)=O)C(C)C1 C1(C(=O)NCC2(C(COC)O)CC2)CCOC1CNC(=O)CCN1CCC1 c1(C(N2CC(CC(C)NC(C3C(C=C)C3)=O)C2)=O)cn(C2CC2)nc1C c1(OC)ccc(C(=O)NC2CC2CNC(=O)COCCN(C)C)nc1.C(C)=O C1(CC)CCN(C(c2cccc(C)n2)=O)C1CNC(=O)COC1CCC1 C12(CNC(C3CC3C(N)=O)=O)CC1CN(C(c1cnn(CC(F)F)n1)=O)C2 C1(c2nnnn2CC2CC2)(Nc2cc(Cl)ncc2)CCCSCC1 N1(C(C(=O)NCC)=O)CCN(C(=O)CCc2cc(SC)c(C)o2)C1C1CC1 c1(C(N(COCC)CC)=O)cc2c(OC)c(OC)ccc2[nH]1 C(=O)(CCS(=O)(=O)c1ccccc1)N1C(CNC(CC(C=C)C)=O)C(O)C(O)C1 c12cc(ccc1Cl)CNC2=O.CN1CC(CN2CCN(C3CC3)CC2)CC1=O C(=O)(C1=C(C)N(C)c2ncnn2C1)N1C2(CN(C(C(CCC)C)=O)C2)CCCC1 C12CC(C1(C)C)CC(=O)N2.C(C(C(=O)NCCCn1ccnn1)OC)SCC C1(NC(C(c2ccc(F)cc2)(C)F)=O)CC2CC1N(C(c1scnc1Cl)=O)C2 N1(C(c2c(COC)cccc2)=O)CCCC(NC(c2snc(C)c2N)=O)CC1 c1(C(N2CCC(C(N(C(CCSC)C)C)=O)CC2)=O)sc2ncnn2c1C c1(CC)cc(C(=O)NC2CCCC2CNC(C2(C)CS(=O)(=O)C2)=O)n(C)n1 C1(CN(C(CC=C)=O)CC)CN(C(C2CCC2OC)=O)CCO1 C12(C(=O)NCC3C=CC(NC(C(n4c(C)ccn4)C)=O)C3)CCC(CO)(CC1)C2 C1(CNC(C(CC#C)C)=O)CCN(C(c2cc(C3CCC3)no2)=O)C1(C)C N#Cc1csc(NC(C2CC3CC3N2C(c2cccc(-c3ccsc3)c2)=O)=O)n1 C(=O)(C(C(=O)NCC(C)(O)CNC(c1ccc(-c2cc[nH]n2)s1)=O)C1CC1)OC C(N=c1nc(N2CCC3CC23)c2c(F)cccc2[nH]1)c1ccc(C)nc1C1CC1 C1(O)(CNC(C(CC)Cc2ccccc2)=O)CCN(C(C2COC(=O)C2)=O)CC1 CC(C)CC(C(=O)NCC(CO)NC(c1cn(C2CCOC2)nn1)=O)C(C)C c1(NC(CNC(C(C)=C2CCCC2)=O)C(C)C)ncnc2c1cnn2C(C)(C)C CC1(C)CCN(C(C2CC(=O)N(O)C2)=O)CC1CNC(=O)Cc1cnsc1 c1(C(=O)NCC2CC(NC(c3ncnn(C)c3=O)=O)C2)cc(Cl)cc(Cl)c1N N1(C(c2ccc(COC)o2)=O)CC(NC(C2CC3CCC3C2)=O)CC12CCCC2 N1(C(CNC(C2C(C)C2)=O)=O)CCC(NC(=O)CCOc2ccccc2)CC1C c1(C(=O)NCCC(CNC(c2cccc(OC)c2)=O)O)cc(F)c(N)c(F)c1 N1(C(C(C)NC(CCCOCC)=O)=O)CCC12CN(C)C2 c1(C(=O)NC2CN(C(C3=CCCC3C)=O)CC2C)n[nH]c2c1CCCC2 CC1CN(C(c2ccnc(N3CCCC3)c2)=O)CC1NC(=O)C(O)CNC(N)=O c1(C(C)OC)ncc(C(=O)NC(C)CC(C)NC(=O)CSc2ccccn2)s1 C1(N(C2CCN(CCS(C)(=O)=O)CC2)CC#C)CC12CCCC2 C(=O)(C(C=C)n1ccnc1)N(CC(CC)NC(COCC=C)=O)C n1(CC(=O)N(CCNC(C2CCS(=O)(=O)C2)=O)CC)ccc2ccccc12 c1(C(=O)NC(CN(C(C2(CSC)CC2)=O)C)CC)ccc2c(c1)nc(O)n2C Cc1cc(N2CCC(NC(C3CCC(=O)N3C)=O)C(C)C2)nc(C(C)(C)C)n1 C=CC1(O)CCN(C(C2CC(NC(C3(C#N)CC4CC4C3)=O)C2)=O)C1 C(C1c2ccsc2CCN1C(C1CCCS1)=O)NC(C(C)n1cccn1)=O c1(CC)ccc(C(N2CC(NC(=O)CC3(N(C)C)COC3)C(C)C2)=O)cc1Cl C1(C(=O)NCCc2cnns2)(NC(=O)CC2CCOC2)CCCC1 c1(N2CC3(CN(C(c4c(C)cc(Cl)cc4C)=O)C3)C2)cc2c(cn1)C(=O)CCC2 N#Cc1cccc(CC(=O)NCCN2CCN(C(C3(F)CCCOC3)=O)CC2)c1 C(C(C)(C)CC(=O)N(CC(C)C#N)C)NC(c1c(C)nc(CC)o1)=O N1(C(CSCC(N)=O)=O)CC2CCCC2(C(=O)NC(CC2CC2)C2CC2)C1 C=CC(CCC)CC(=O)NCC1(O)CCCN(C(=O)C=Cc2cn[nH]c2)C1 Cn1c(C2CC2)nn(CC(=O)NCC2CC(NC(C3(C)CC3F)=O)C2)c1=O Cc1cc(NC(=O)C(c2cn(C)nn2)NC(=O)C2=COCC2)c(O)cc1F C1(O)(C(N(C)Cc2ncccc2Cl)=O)CCCN(C(c2ncn(C)n2)=O)C1 C1(CNC(c2c(CC)nc(C)nc2)=O)CN(C(=O)CCC#N)CCC12CCC2 c1(C(N(C)CCC2CCCCN2C(=O)CC2CC3CC3C2)=O)cncc(F)c1Cl c1(CNC(C2C(NC(C=C(C)C)=O)CCC2)=O)cnn(C)c1O C1(NC(=O)Cc2cc(F)ccc2O)CC1C1CCN(C(c2ccc[nH]2)=O)CC1 N1(C(c2ncn(C(C)C)n2)=O)CCC(CC(=O)NCCCOc2ccsn2)CC1 c1(C(N2CC(NC(=O)C(F)C3CCC3)CC(C)C2)=O)ccc(Cl)c2occc12 c1(C(=O)NCC(c2ccccc2)N(C(C2C(=C)C2)=O)C)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2c(O)ccc(C)c2)=O)CC(NC(c2coc(Cl)n2)=O)C12CCOCC2 C1(CNC(CC2(OC)CC2)=O)CCNC(C)C1 c1(C(N2CC(NC(c3cncnc3)=O)C(F)C2)=O)n[nH]cc1[N+](=O)[O-] N1(C(C(=O)NC2(C)CCCC2)=O)CCC(NC(C2CCCN2N=O)=O)C1(C)C C(c1ccc(F)cc1)=C(C)C(=O)OC1CC2CC(C(=O)OC(C)(C)C)C2C1 C1(C(=O)NC2(C)CC(=C)C2)CCN(C(=O)CCCC#CC)O1 c1(CNC(C2COC(CO)C2)=O)ccc(CNC(C2(F)CC=CC2)=O)cc1 Cc1cc2[nH]c(C(=O)NC(C)CCNC(C3(C)CCC(C)C3)=O)cc2o1 Cc1nc(C(N2CC3CC2CN3C(c2ccc(I)cc2Br)=O)=O)ccc1F c1(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)C)ccnc(-n2cccn2)c1 CC1CNC(=O)C1.C1(C(=O)NCC(C)(C)CN(C)C)OCCC1(C)C c1(C(N(CC(O)CNC(=O)Cc2ccccc2)C)=O)ccc(CCO)cc1 CCC(CC(F)(F)F)C(=O)NC(CCN(C(=O)C(CC)CC)C)C(C)(C)C c1(C(N2C(CCNC(=O)C3CC3)CCC2)=O)cc(CO)ccc1Cl c1(C(=O)NC2CCN(Cc3ccc(O)cc3F)C2)c(F)ccc(Cl)c1Cl C(=O)(CC(C(F)F)NC(=O)C(C)OCCC(C)C)N(C(C)COCC)CC Cc1cnc(Cl)c(C(=O)NCC2CN(C(c3cccn3C(C)C)=O)CCO2)c1 c1(C(=O)OC)ccc(Cl)c(NC(C2CCC(NCc3ccncc3O)C2)=O)c1 CC1(CCNC(c2conc2CNC(c2cscn2)=O)=O)CCCO1 N1(C(C(CC2CCC2)OC)=O)CCC2(CC(C(=O)NCCC3CCCOC3)C2)C1 C(=O)(C(F)(F)C(O)C1CC1)C(C1(C(=O)NCCC2CN(CC)CCO2)CCC1)=O c1(C(=O)OC)ccc2ncc(CNC(=O)Nc3nc4c(s3)CCC4)n2c1 C(=O)(C(C1=Cc2ccc(OC)cc2OC1)N1CCC(OC2CC2)C1)NC(CC)C C#Cc1cccc(CC(=O)N(CCCNC(=O)C=CC=CC)C)c1.N CN1CCCC1C=CC(=O)N(C1CCSC1)CCNC(=O)CNC=O c1(CNC(=NCCC(C)C)NCc2ncnn2C(C)C)cc(F)c(N)cc1F C(=O)(NNC(=O)C(C)SC1CCCC1)c1cc(OC)c(C(C)(C)C)cc1 Nc1c(C(=O)NCC2(F)CCN(C(C3CC34CCCC4)=O)C2)ccc(F)c1F C=Cn1ccnc1C(c1nnnn1CCOC)NC(C1(C)CC1(C)C)C1(C)CC1 c1(C(=O)NC(C(C)NC(C2CC(CCC)C2)=O)C)ccc(N(C)C(C)=O)cc1 c12ccc([N+](=O)[O-])c(c1)OOC2.c1(OCC)cccc(CCc2ccccc2)c1 C1(C(C)NC(C2(COC)CCCC2)=O)CCCN(C(c2nn(C)nc2C)=O)C1 N1(C(c2c(OC)ccs2)=O)CCCC(C)(C)C1CNC(C1(S(C)(=O)=O)CC1)=O C12(NC(c3nc(CC)oc3)=O)CCC1CN(C(C1(C)C=CCCC1)=O)C2 c1(C(=O)NC2C(OC)CN(C(C3(O)CC3(C)C)=O)C2)nn(C)cc1S(C)(=O)=O C1(C(=O)NCC2CCN(C(CN(CC)CC)=O)C2)CCc2nc[nH]c2C1 Cn1ncc2cc(C(N3C4CCC3CC(Nc3ncncc3I)C4)=O)ccc12 Cc1cc(C(=O)NC2CCCCC2CNC(c2ccnn2C)=O)cnn1 N1(C(C(=O)NC)C2(C(=O)OC(C)(C)C)CC2)CCn2c(cnc2C(N)=O)C1 c1(C(N2C(CC)C(NC(=O)C(C)OC)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 N1(C(C=C(CC)C)=O)C2CCC1C(F)C(NC(=O)Cc1c(Br)cnn1C)C2 c1(C(=O)NCC2=CCCN(C(C3CC4CCC3C4)=O)C2)cccc2c1C(=O)CC2 C=CC(C)C(=O)NC(CN(C(=O)CCc1cnn(C)n1)C)CC c1(C(N2CC(N(C)C(C3(c4ccccc4)CC(F)C3)=O)C2)=O)ccc(O)cn1 C1(CNC(CN(C(C)=O)C)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)C12CC2 c1(C(=O)NC(CNC(CN(CCOC)C)=O)C(C)C)ccc2oc(C)nc2c1 N1(C(CC2CC(OC)C2)=O)CCN(C(c2cccc(-n3cncn3)c2)=O)C2CC12 C=CC1CCCC(NC(C2(C)CCCN2C(=O)CCCCCOC)=O)C1 O=C1CCC(CC(=O)NC2(C(=O)NCCC3COCC3O)CC2)CN1 N1(C(c2cnc(CC)nc2C)=O)CC2CC(NC(=O)C(C)(C)C(N)=O)C(C2)C1 C(=O)(CN=c1[nH]cnc2ccc([N+](=O)[O-])cc12)N1CCCc2ccccc21.CC(C1CC1)SC CC1(CC(=O)NCCN2CC3CC3C2)CCN(C(=O)C2=CCSC2)C1 C1(C(=O)NC2CCN(C(c3nnn(C)n3)=O)C2)CC2(CO1)CC(F)(F)C2 N1(C(c2c[nH]c(Br)c2)=O)CCC2(CCN(C(=O)CC(O)C3CC3)C2)C1 c1(CC(=O)N(C2CCN(C(C3CCC(C)(C)C3)=O)CC2)C)ccc2c(c1)OCO2 C1(NC(CC(=O)NCC#C)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)C12CCCC2 c1(CN(C)CCNC(c2nn(-c3cccc(Cl)c3)cc2O)=O)ccc(C#N)cc1 N1(C(C2CCC(C(N)=O)O2)=O)C2CCC1CN(C(=O)CNS(=O)(=O)C1CC1)C2 N1(CC(C)C)CCCCC(NC(=O)C(N2Cc3cnn(C)c3C2)=O)C1=O C1(C2CN(C(=O)CC3CC4(CC4)C3)C2)(NC(c2cnc(C(F)F)nc2)=O)CC1 Clc1cc2nc(N3CCN(Cc4ccns4)CC3)ccn2n1 n1(CCS(N)(=O)=O)nc(CC2CCOCC2)nc1-c1cnn(CCF)c1 C1(CC(=O)NC2CCC(C)(CNC(C3(CO)CCCO3)=O)C2)NC(=O)NC1=O C1(C(=O)NC(CC=C)CNC(c2cccn2C2CC2)=O)CCCN2CCCC12 N1(C(C(C)NC(CC)=O)=O)C2CCCC1CN(C(=O)C(O)CC(C)C)C2 CN1CC=C(CC(=O)N2CC3CCC2(CNC(=O)C=CC2CCOC2)CC3)CC1 N1(C(c2cc(CCOC)on2)=O)CCC(O)(CNC(C2(C)COC2)=O)CC1 c1(OC)ccnc(C(N2CCC(NC(C3CC3F)=O)C2c2ccccc2)=O)c1F C1(CCC(=O)N(CCCC)C(C)CC)CCCCN(C(=O)CCCOCCOC)C1 c1(SCCC)cc(C(N2CC(CNC(c3csc(=NC)[nH]3)=O)C(C)C2)=O)ccn1 Cc1nc2c(s1)CCCC2C(=O)NCCC(C)(C)NC(C1CC(C#N)C1)=O C(=O)(C(C#N)C(C)(C)C)N1CC(CC(C)NC(C2(CC)CCCCO2)=O)C1 C1(CC(=O)NCC2(O)CC(NC(C3CCN(C(C)=O)C3)=O)C2)CCCC12CC2 c1(C(c2ccco2)=O)ccc(-c2nc(-c3cc(C4CC4)no3)no2)s1 C=C1CC2(C1)CC(C(=O)N(CC(C)NC(=O)CCN1CCC(C)CC1)C)C2 C(=O)(C(C)(CC1CCC1)OC)NCCN(C(C1CCCN1CC)=O)CC C(=O)(CCCCCc1cccs1)NCC1(F)CCN(C(c2cc(OC)n[nH]2)=O)C1 c1(OC)cc(CN2CCOCC(NC(c3cnc(Br)s3)=O)C2)ccc1I c1(COC(=N)O)cn(CCCC(=O)N2CCCC2CC2CCOCC2)nn1 C1(C(N2C(CC=C)CCCC2)=O)CCCCN(C(=O)C(=O)NCC)C1 CC(C)CS(=O)(=O)N(C)C(C1CCN(Cc2ccc(C(=O)O)cc2)C1)=O C(CN=c1ccnc(C2CCC2)[nH]1)N(C(c1cn(-c2ccccc2)cn1)=O)CCO CC1COCC(C(=O)NCc2c[nH]nc2C(=O)NCC2(C)CSC2)O1 c1(C(=O)Nc2cccc(NC(C3CCC(C)(CC)O3)=O)c2)cc(Cl)ncc1O CCC(CCC(=O)NCC12CC(CC)(CN1C(=O)CC1CCSC1)C2)OC N1(C(C(C=CCCC)O)=O)CC2CCC1CC2NC(c1csnc1Cl)=O C=C(CNC(=O)CC1CCCN1C(=O)C(C)S(C)(=O)=O)c1ccccc1 C1(C(=O)NCCN(C)CC)CCC(CC)C1.c1(C(=O)N)coc(C(=O)OC)n1 c1(CNC(C2CCCN(c3ccccc3)C2=O)=O)cc2ncsc2o1 c1(C(=O)NCC2(NC(CC(C)NC(N)=O)=O)CC2)cccc2c1S(=O)(=O)CCC2 c1(C(N2CCC(C)C2CNC(c2c[nH]nc2[N+](=O)[O-])=O)=O)cc(F)cc(N)c1F c1(C(N2CCC(NC(C(CC)(C)OC)=O)C2)=O)ccc2c(c1)nnn2C CC1(O)CN(C(C2CCC(C3CC3)N2C(=O)CCCn2cncn2)=O)CCC1O c1(-c2c(F)ccc(OCC)c2)cc(C(N2CC(O)CC2(C)C)=O)c2cn[nH]c2c1 CC1(C)CCC1CC(N1CCC(N2CCC2)CC1)=O.C(=O)(C=CCO)NCCO C1(NC(C(c2ccnn2C)C)=O)CC2(C1)CN(C(=O)Cc1cscn1)C2 C1(C(=O)NC2CCN(CCC)C2)CC(C)CN1C(c1c[nH]nc1C(C)C)=O C(=O)(CCC(=O)c1ccc[nH]1)N1CC(C)(NC(=O)Cn2cc(Br)cn2)C1 N1(C(C(C)N(C(=O)CCc2ccncn2)C)=O)CC(O)CC1(C)CO CC1(C)COC(CNC(=NCCF)NCc2ccc(F)nc2)=N1 c1(CC(=O)NC2CC3CC(NC(c4cc(F)c[nH]4)=O)CC23)c[nH]c2ccccc12 N1(C(C=C2CCC(C)CC2)=O)CCc2ccc(Cl)c(F)c2C1C C1(NC(C2(C)CN(C(CC(=O)NCC#C)=O)C2)=O)CCOC12CCCC2 C1(C(N(CC=CC(=O)NCCC(=O)NC(C=C)C)C)=O)CCCC1OC CCC(COC)(CC)C(=O)N1CCC2CC12C(N1CC(C)OC(C)C1)=O C1(NC(=O)CCNC(C(C)CC2CC2)=O)CCN(CCO)CC1.CC(C)(C)CO Nc1cc(C(N2CCC(NC(C3CCCCCC3)=O)C23CCC3)=O)cc(F)c1O c1(C(C)(C(=O)OC)OC)ccc(C(=O)NCC(O)CC2CNC2)cc1 N1(C(C2CC(OC(F)F)C2)=O)CCc2cc(CNC(C3CC(O)C3)=O)ccc2C1 S(=O)(=O)(c1ccccc1Cl)NCC(=O)NCCN(C(C1CC(=O)N(O)C1)=O)CC CCC(CC)CC(=O)NCC(C)(C(C)C)NC(c1cn(-c2ccccc2)nn1)=O C(=O)(CCC(C)(F)F)NCC(CNC(C(CC)n1ccnc1)=O)O C1(C)(C(N(CCN(C(=O)CC2CC(C)(C)CO2)C)C)=O)CNC(=O)N1 c1(C(=O)NCC2CCC(NC(CC(=O)OCC)=O)C2)c(Cl)cccc1Cl C1(NC(c2[nH]cc(CC)n2)=O)CN(C(=O)C(n2ccc(C)n2)C)CCC1CO c1(C(=O)NC2C(C)N(c3nc4cccc(F)c4s3)CC2)c(Cl)ccc2c[nH]nc12 CCS(=O)(=O)CC(=O)NCC1(CNC(=O)CCN(C)CCO)CC1(F)F C1(C(=O)NCC(CNC(C2(COC)CC=CC2)=O)(C)C)CCS(=O)(=O)N1 C1(C(=O)OC)CC(F)CN1C(C12CC(CO)(C1)C2)=O.C12CC3CC3N1C2=O CCCCC(CC(=O)NC1CC(O)(C(F)F)C1)NC(=O)CC(C)N(C)C c1(CN2C3C=CCC2CCC3)ccc2n[nH]c(C)c2c1.Cc1c2ncnc1NC2=O N1(C(C=Cc2n(CC)ccn2)=O)CCC(C2(NC(c3ncccc3F)=O)CC2)C1 c1(NCCCCS(C)=O)ccc(S(=O)(=O)N2CCOc3ccccc3C2)c(Br)c1 N1(C(c2cc(COC)no2)=O)CCOCC(NC(c2ccc(O)nc2Cl)=O)C1 C1(C(=O)NCC(c2cccs2)C)C=CCN1C(c1cccs1)=O c1(C(=O)NC(CCC=C(C)C)C)cccc(CNC(c2cncc(C)c2)=O)n1 C1(CCNC(C2(N(C(c3cnc(SC)s3)=O)C)CC2)=O)CC2CCC1O2 N1(C(C2(C#N)CCCO2)=O)C(C(=O)NCCC2=CCCCC2)CCC12CC2 Cc1nc2ccc(C(=O)NCC3(F)CN(C(=O)C(C#N)C(C)C)C3)cc2s1 c1(CSC)noc(CC(=O)NCCC2CCN(C(C3CC(C(F)(F)F)C3)=O)C2)n1 c1(C(N(CC(CN(C(=O)CP(C)(C)=O)C)O)C)=O)ccc(C(F)(F)F)nc1O C1(NC(c2nc(C)[nH]c2Br)c2n(C(C(=O)OC)C)nnn2)CNC(=O)C(F)(F)C1 c1(COCC(=O)NC(C2CCCO2)Cc2ccccn2)ccccc1F c1(CN2C3C(C#C)CC(CC3)C2)c(-c2ccccc2)nc2cc(Cl)ccn12 N1(c2nccc(C(C)C)n2)CCC2(CC1)CN(C(=O)C(F)(F)C(C)(C)O)CCO2 CC(C)C(C(=O)NCCN(C1COC1)C(C1CCCC1)=O)c1cccnc1 c1(C(=O)NC2CCCCN(c3nnc(CCC)s3)C2)ccc2c(c1)nnn2CC c1(CN2CCCC(C(=O)NC(c3ccccn3)CO)C2)ccc(O)cc1O c1(C(=O)NC2CC(C)N(C(=O)C(c3ccncc3)C)CC2)cccc2ccsc12 CC1(c2ccccc2)CCCN(N2CCC(NCc3ncccc3Br)C2)C1 CC1CCN(C(c2ccc(Cl)cc2)=O)C1C(N1CC(C2CCCO2)C1)=O c1(C(N2C(CN(C(CC3C(C)C(=O)CC3)=O)C)CCC2)=O)ccn2cncc2c1 C1(CC(=O)N(CCNC(C(C)NC(N)=O)=O)CC2CC2)CCC(C)(C)O1 N1(C(C(C(C)C)C2CCC2)=O)CC2(C(=O)NC(C)C(F)(F)F)CC1CO2 N1(C(CC(C(C)C)C)=O)CCCC2(CCCN2C(c2cnc(Cl)s2)=O)C1 CN1CCC(C)(C(N2CCCC(C(=O)NC3CC(F)(F)C3)C2)=O)CC1 C(=O)(CC1=CCOCC1)OC.CC1CCN(C(=O)CCCCNN2CCCC2)CC1 c1(COC(=O)CCC(O)Cc2nn[nH]n2)ccc2c(c1)OCO2 C1(C(N2CC(CC3CC3)C2)=O)CC2(CCN1C(=O)C=Cc1cccnc1)CC2 C(c1cn(C)cn1)=CC(=O)NCCCN(C(C=CCC)=O)CC1CCCC1 c1(C(=O)NC(C)CC2CN(C(C3CCCCC3(F)F)=O)C2)cc2c([nH]1)CCC2 Cc1nn2cc(C(=O)NC3CCCC3NC(c3ncoc3C)=O)nc2s1 c12ccccc1C1CCCC1NCCCO2.c1(OCC)sc(C)cc1OC C1(C(=O)NC2(CC=C)CCN(C(C3CC4(C3)CC(C)C4)=O)C2)CCC2(CCC2)C1 N1(CCC(=O)NC(C)CN(C)C(c2ccc(C(F)F)o2)=O)CCCCC1=O Cc1cc(C(=O)NC(C)C(=O)NCc2sccc2C)ccc1O C=CC1(NC(C2(COC)CC(N)C2)=O)CCC1 N1(C(C2(NC(C)C)CC2)=O)CC2CCCC(C1)N2C(=O)C(F)Cc1ccccc1 C12(SCCCNC(CC=C)CC)CN(C(=O)OC(C)(C)C)CC1C2(F)F c1(C(=O)NC(C2(O)CN(C(c3cc(C)c(F)nc3)=O)C2)C)cccc([N+](=O)[O-])c1 C1(C(=O)NCC2(C(=O)NC(C(C3CC3)OC)C)CCCO2)CCC(C)CC1 Cn1ncc(C(=O)NC2CC(C(F)C(N3CC4CCC4C3)=O)C2)c1C#N Cc1cc2ccc(C(=O)N(CC(C)CNC(C3(CF)CCC3)=O)C)cn2c1 N(C1CCCc2cnn(C(C)C)c21)C(=O)Nc1c(C)nc(C(N)=O)cc1 c1(NC(CC)=O)cccc(C(=O)N(C2CN(C(=O)Cc3cc(Cl)no3)C2)C)c1 C1(NC(CCOCCCOC)=O)CC12CCN(C(c1c(C)cccc1F)=O)CC2 CN1CC(C)(C(=O)NCC(O)C(=O)NC2CCOCC2F)CC1=O C1(CC=C)(NC(c2cn(C(C)C)nc2C)=O)CCN(C(=O)CSCCOC)C1 C1(CCC(=O)N(C2CCC2)C2CC2)CCN(C(c2ccns2)=O)C1 N1(C(CC2C(C)(C)N(C(C3COC(=O)N3)=O)CC2)=O)CC2COCC2(C#N)C1 c1(C(=O)NC2CN(C3CN(C(C4(C#C)CC4)=O)C3)C2)cc(F)cc2cnccc12 Cc1cnc(CN2CC(CNc3ccnc(-c4ccc(Cl)cc4)n3)C2)c(F)c1 c1(C(=O)NCC2COCCN2C(c2cc(CO)[nH]n2)=O)ccc2c(c1)OCCN2 N1(C(Cc2ccc(SC)cc2)=O)CCCC(N(C)C(c2ccncc2Br)=O)CC1 c1(C(=O)NCC(C2CCCN(C(c3cnc(C)[nH]3)=O)C2)(C)O)cnc2[nH]cnc2c1 c1(C(=O)NC(C2N(C(C(F)=CC)=O)CCC2)C)ccc(C(=O)NC)nc1 C1(c2nnnn2C2CCOCC2)(NCC2CCCCC2)CCN2CCCCC12 c1(NC(C2(NC(=O)C3=CCCS3)CCOC2)=O)cccc2[nH]ccc12 Cc1nc(C)c(C(=O)NCC2(O)CC(NC(C3CC3C(C)C)=O)C2)[nH]1 CC(CC(F)F)C(=O)N1CCCC1C(C)(C)NC(=O)C(C)C1(O)CCC1 C1(C(=O)NC(CNC(CCC(=C)Cl)=O)(C)CC)CC12CCCCCC2 c1(C(N(CCC(C)NC(C2(CCCC)CC2)=O)C)=O)cccc2c1NCC2 N1(CC)C(=O)CCC1C(=O)N(C)CC1(O)CCN(C(=O)CNS(=O)(=O)NC)C1 C(C(=O)NCC1COCCN1C(=O)CC1(C)CC1)(C(C)(C)C)SC c1(C(=O)NC2CN(C(CCCN(C)C)=O)CC(O)C2)ccc2c(c1)C(C)(C)CO2 c1(C(=O)OC(CCC)C(=O)OC(C)(C)C)ncccc1C#N C1(N(CC#C)C(C2CC2C=C)=O)CCCN(C(=O)Cn2ccc(C(F)F)n2)C1 C(C(CC(F)(F)F)NC(c1ccnn1C)=O)NC(C(C)OC)=O N1(C(C2(CNC(C=CC)=O)CCCO2)=O)CCCCCCC1C Cc1[nH]nc2ncnc(CNC(=NCc3ccc4c(c3)OCO4)NC(C)C)c12 N1(CC)CC(NC(CC2CCN(C(c3cncnc3C(C)C)=O)C2)=O)CC1=O N1(C(c2cccc(C#C)c2)=O)C2CCCC1CC(NC(C13CSC(C1)C3)=O)C2 C1(CNC(C(CC)n2ccnc2)=O)CN(c2cc(OC)ncn2)CCCO1 C1(C(N(C(C)C)CCN(C)Cc2cc(Cl)sc2Cl)=O)CC2CC2CC1C N1(C(CC2CC(C)C2)=O)CCN(C2CCCN(C(c3cscn3)=O)C2)CC1 C1(CC)CN(C(=O)Nc2ccc(Cl)c(OC)c2)CCN1Cc1ccccc1C C(CC(F)F)(C(=O)NCc1cnc(O)nc1O)NC(C(COCC)C)=O C1(CNC(NCC2CCCC(OCC)C2)=NCC2CC2)CCS(=O)(=O)CC1 N(C1CCc2ccccc21)C(C1CCCN(C(=O)C(=O)NCC(F)F)CC1)=O Cc1c(N)ccc(C(=O)NC2CCCCN(C(c3cc(C(N)=O)c[nH]3)=O)C2)c1F N1(C(C(CC)CC)=O)CCC(C)(C)C1CC(=O)NCCOC1CCCC1 N1(C(CCCC=C)=O)CCC2(CCN(C(c3cccc(COC)c3)=O)C2)C1 n1(CCCC)cccc(C(N2CC3CC(NC(c4cnc(C)[nH]4)=O)C2C3)=O)c1=O CC1C(NC(c2ccc[n+]([O-])c2)=O)CC2CCC1N2C(c1cn(C)nn1)=O C=C(C)CCCC(=O)NC1COCCN(C(C2COCCOC2)=O)C1 c1(C(=O)NC2C3CN(C(C(=O)NC4CC4)=O)C2C3)ccc2nc(Cl)nn2c1 N1(C(CSCCCC)=O)CCC(NC(c2oc(CC)cc2C)=O)C(C)C1 C1(CC(=O)NC2CN(C(CC(C)CN(C)C)=O)C2)CC2(CCOCC2)CO1 C1(OC)CC2(C1)CC2NC(c1cnn(CCNC(C2(CC(C)=O)CCC2)=O)c1)=O N1(C(c2ccc(F)c(OC)c2F)C(=O)NC(C)(C)C)CCC2COC(=O)NC2C1 N1(C(c2c(F)ccc(C)c2)=O)CC(NC(=O)C(F)CC2CCCC2)CC12CCC2 C(=O)(C1=CC2CC(C1)CC2O)N(C1CC1)CC1N(C(c2cc(C)ns2)=O)CCC1 N1(C(c2c(C)ccs2)=O)CCCN(C(C2COC3CCCCC23)=O)CC1C CC1=NOC(C(=O)NC2(C)CC(C(=O)NC(C)Cc3nc[nH]n3)C2)C1 C1(C(=O)NCCn2ccnc2C)(CC)CN(C(c2cc(O)cs2)=O)C1 C(=O)(C1=CCCN(C(=O)C(CO)OC)C1)N(CC=C)CCO C1(NC(C2CC(CN(C)C)C2)=O)CCCCN(C(C2CC(=O)CCO2)=O)C1 c1(C(N2CCC(CNC(C(CC)C)=O)C2)=O)cc(Cl)cc(C)c1OC Cc1[nH]nc(C(=O)NC(c2nccs2)C)c1Br.N12CCC(C1)C2=O N1(C(CCCCC#C)=O)C2CC=C(C(=O)N3CCC3=Cc3ccccc3)C1CC2 c1(OC)ccc(C)c(C(N2CCC(NC(=O)C3CC3)C2)C(=O)NC(C)C)n1 CCCC(C(=O)NCC1C2CN(C(=O)CSCc3cccc(C)c3)CC12)C(C)C c1(NCC(C)NC(CCc2c(C)cccn2)=O)ncnc2c1c(Br)nn2C c1(C(=O)NC2CCCN(C(C3C(C)OCCC3)=O)C2)c(F)ccc(F)c1N C1(C(=O)NCC(C)(C)N2CCCC2)CC(NC(C2CCCCC2O)=O)C(O)C1 C(=O)(C(F)(F)C(F)(F)F)NCc1nccc(OC2CCN(C(C3C(=C)C3)=O)C2)c1 N1(C(CNC=O)=O)CCC2(CCCN2C(=O)CNC(C2CCS(=O)(=O)C2)=O)C1 N1(C(Cc2cc(OC)no2)=O)CCCCCC(NC(c2ccc(F)cc2O)=O)C1 C(C(C)C(C)C(=O)NCCOC1CN(C(c2ccc(=O)n(CCF)n2)=O)C1)OC c1(C(N2CC(NC(C(COC)O)=O)C(CO)CC2)=O)c(F)cc(Cl)cc1F N1(C(c2cc(C)oc2)=O)CC(C)(C)CCC1CNC(=O)CCCn1cccc1 CP(C)(=O)CCc1ccc(C(N2CCCC2CNC(=O)CC2CC(CF)C2)=O)s1 c1(C(C(=O)NCCOCCN(C)C(C2(C)CC2Br)=O)C)cnc2ccccn12 c1(N(C2CC(F)CN(CC)C2)C(c2ccc(Cl)cc2)=O)ccc2nonc2c1 c1(C(N2C(C)C(NC(=O)CC3(O)CC3)CC2)=O)cc2cc(Br)ccc2[nH]1 C1(NC(N(C2CC2)CC)=O)CC(NC(N)=O)C12CCC2.c12ccc(o1)CNC2=O c1(OC)ncc(Br)c(=NCC2(NC(c3ccnc(F)c3Cl)=O)COC2)[nH]1 c1(OCC)cccc(C(=O)NCCCCNC(=O)Cc2cccnc2C)c1 c1(NC(N2CCCc3cc(Br)ccc32)=O)cnc2c(c1)C(=O)NCC2 C1(C(=O)NC2C(NC(CCC=CC)=O)CCCC2)CCCC2(CC2)C1 N1(C(CNC(c2c(C#C)c[nH]n2)=O)=O)CC(C2CC2)(C(=O)OCC)C1 C1(N(C(CC=CCC)=O)C)CCCC(NC(c2cnc(OC)cn2)=O)C1 C12(NC(C(C)NC(C)=O)=O)CCC(CNC(C3CCC(C)(C)CO3)=O)(CC1)C2 CC1(C)CCN(C(C)=O)C1CC(N1CCC(C)(F)C1)=O.C(=O)CCc1nc[nH]n1 N1(C(=O)C(F)F)CCCC1C1CCCN1C(c1cc(CF)on1)=O C(=O)(CC(C)(C)C(F)F)NC(C)CCC(N1CCOC(C)(C)C1)=O n1(CC(N2CC(CNC(C(C)=CC)=O)CC2(C)C)=O)cc(C#N)c(O)nc1=O C(=O)(C(CC)(CC)CC)N(CCN(C(=O)C=Cc1cc[nH]n1)CC)CC n1(CC=C)cc(C(=O)NCC2CCCN2C(=O)CCCOCCC)nn1 N1(C(c2nc(CC)[nH]n2)=O)CCC(C(F)(F)F)C(NC(=O)CC2CC(C)=NO2)C1 C1(NC(COCCC)=O)CN(C(c2cc(-c3ccn(C)n3)on2)=O)CC1O C=CC1(CC(=O)NCc2cc(Cl)no2)CN(C(=O)C=Cc2cscn2)C1 Cc1cc(CNC(=O)C(CC(F)F)NC(=O)CC(Cl)Cl)cc(O)c1 C1(NC(C(C)Cn2cccn2)=O)(CO)CCCN(C(C2(CO)CCCO2)=O)C1 CC1=C(C(=O)N2CCC(C(C)NC(c3cnnc(Cl)c3)=O)C2)CCO1 Cc1cc(C(N2CC3CC(NC(c4cnn[nH]4)=O)C2C3)=O)cc2c[nH]nc12 c1(C(C)NC(C(=O)OC)(C)CC)cc(I)ccc1Br c1(CN2CCC3(C(C(=O)NCCCO)C3)C2)cc(Br)cc(Br)c1F Cc1cc(NC(C2(C(F)(F)F)CCC(O)CC2)=O)c(C)cc1F C1(C(N2CC(CCC)N(C(=O)COCCOC)CC2)=O)CS(=O)(=O)CC12CCC2 C1(NC(c2n(CC)ncc2Cl)=O)Cc2ccccc2C1NC(=O)C=C(C)C1CC1 CN1CC=C(CC(=O)NC(C2CCOC2)CNC(c2cnc[nH]2)=O)CC1 CCCCCC(O)C(=O)N1CC(C(O)C(=O)NC2CCC(C)(C)CC2)C1 C1(CC(N2C(C(=O)NC3CCS(=O)(=O)C3)CCCC2)=O)CCC(F)(F)CO1 Cc1cc(C(N2CCC(NC(=O)C=CC3CCOC3)C23CC3)=O)c(C)c(C)c1 c1(NCC(C2CC2)NC(c2ccc(C)cc2Cl)=O)ncnc2onc(C)c12 c1(CCC)n[nH]cc1C(N1CC(CC(C)NC(=O)C=CC2CCOC2)C1)=O CC1CN(C(=O)C(C)(C)C(N)=O)CC(C)C1NC(=O)CSC1CC1 CCCCC(O)C(C)C(=O)N1C2CCC(C2)C1C(=O)NC1CC(C(C)O)C1 N1(C(C(CCCC)C)=O)CC(NC(=O)CNC(=O)NC)CC2(CC2)C1 C(=O)(C#CC1CCOCC1)NC1CC(CNC(c2ccc(SC)cc2)=O)C1(C)C N1(C(c2cc(C)nc(O)c2)=O)CC2(CCC(C(=O)NC3CS(=O)(=O)C3)O2)C1 c1(C(=O)NC2C(NC(C3CN(CC)C(=O)C3)=O)CCCC2)ccc(F)c(Cl)c1 C1(NC(C2CCC=CCC2)=O)CN(C(c2ccc(CCC3CC3)cc2)=O)C2CC12 c1(NCC#N)cc(=NCC2CCCCC2c2ccc(Cl)cc2Cl)[nH]cn1 C1(NC(C(N(C(CC(=O)OCC)=O)C)C2CC2)=O)CCC(=O)N(C)C1 C=CCC(CC(C)C)C(=O)N1CCC(OCC(N2CC(N3CCOC3=O)C2)=O)C1 C1(CNC(=O)OC(C)(C)C)CC(C(=O)NCC2COCC2C(F)F)CC1O.C C(CCN(C)C(c1c[nH]nc1C(C)(C)C)=O)(C(C)(C)C)NC(C(CC#C)C)=O C1(COC)CN(C(c2ncc(N)cc2Cl)=O)CCN1C(=O)C(C)OCC(C)C C1(NC(c2nc(C)oc2)=O)CC2CCC1N2C(c1ccncc1N)=O C12(NC(CC(CC)OC)=O)CCC(F)(F)CC1CN(C(=O)CN(C)CCO)C2 C#CC1(O)CC(C(=O)NC2CN(C(=O)C(C)Oc3cccc(Cl)c3)C2)C1 c1(OCCN(C(C(=O)NC(C)Cc2nccn2C)=O)C)ccc(F)cc1 NC1CCC2C(C(c3nnnn3C3CCC3)NC3CC3)CCC12 NS(=O)(=O)c1n[nH]cc1C(=O)NCCCC1CCN(C(C2CCCC2O)=O)CC1 Cc1c(C(N2CC3CN(C(=O)CNS(C)(=O)=O)C3C2)=O)cc(F)cc1[N+](=O)[O-] Cc1nc(C2CC2)ncc1C(=O)NCC(C)(C)CCNC(=O)Cn1cncn1 C1(C(=O)NC(CC=C)CNC(C2CC2c2ccnn2C)=O)CCC(NC(N)=O)CC1 c1(C(=O)NCC2(C(N)=O)CN(C(C(CCC)O)=O)C2)nc(OC)ccc1[N+](=O)[O-] C1(CC)CCCC(CNC(C2CCOC2CNC(c2cnc(S)nc2)=O)=O)C1 C1(NC(c2c(C)scc2)=O)CN(C(=O)C=CBr)C2(CCCOC2)C1 c1(C(=O)NC(C(=O)NCC2N(CC)CCCC2)CCC2CC2)ccc(C#N)cn1 C12CCN(CC1)C(c1cnc[nH]1)C(=O)N2.C1(C(=O)NCC#C)CCCCC1 C1(CC=C)COCC1N(C(c1nnn(C)n1)C(=O)NCc1ccco1)C c1(C(=O)NC(CNC(C2CCC(C(C)(C)C)O2)=O)C2CC2)cnn2c1OCCC2 Cc1ccc(O)c(C(N2CC=CC2C(=O)NCC(=O)NCCO)=O)c1 C1(NC(CN(S(CC)(=O)=O)C)=O)COCCN(C(c2cnc(Cl)c(Cl)c2)=O)C1 c1(C(=O)NCC(CC(=O)NC(C#C)CC(C)C)C)ccn2nccc2c1 c1(C(=O)NCCN(C(=O)C(C)SC(F)(F)F)CCOC)[nH]ccc1C1CC1 CN=c1[nH]c(=NCc2nc(C3CCOCC3)cs2)[nH]c(=NCC(C)CCO)[nH]1 C1(NC(=O)CN2CCOCC2)CC2CC(NC(=O)C(Cl)=CCl)C2C1 c1(N2C(CNC(c3cc(CC)n(CCO)n3)=O)CC2)ccc(Br)cc1[N+](=O)[O-] c1(C(N2CC(CCNC(C3C(CC)C3)=O)C(C)C2)=O)cnc2c(c1)nnn2C O=C1CCC2(C(=O)NCCCNC(=O)CCCn3ccccc3=O)CCCC2C1 c1(NC(C(=O)NC(CNC(CC(C)OC)=O)CO)=O)cc([N+](=O)[O-])ccc1C CCC(CC)(CCNC(C1CCCCC1C(F)(F)F)=O)NC(C1CC12CCC2)=O c1(NC(c2cn(CC3CC(NC4CC(=O)C4)C3)nn2)=O)cc(O)nc(O)n1 N1(CC=C)CCC(CN(C(=O)Cc2cc(C)[nH]n2)C(C)=O)CC1 c1(C(N2CCC(C3CCCN3C(=O)C(C)=CC3CC3)C2)=O)ccc(CO)cc1F C1(CC)(NC(=O)CCc2ccn(C)n2)CCCN(C(C2CC2c2cnc[nH]2)=O)C1 C(=O)(NNc1nc(C(=O)O)ccc1C)c1ccnc2ncc(OC)nc21 N1(C(c2ccc(NC)cc2)=O)CC(NC(C23CC2COC3(C)C)=O)C2CC2C1 c1(CN2C3C(C(N4CCCC4c4ccc(Cl)s4)=O)C(C3)C2)cc(Br)cc(Br)c1 N1(C(C2CCCC2OCC)=O)CCC(NC(C2C(=C)CC2)=O)C(C(N)=O)C1 CC1CN(C(C2(c3cccc(F)c3)CC2)=O)CC2(CC2)C1 c1(OC)ccc(C(=O)N(C2CCCC2O)C)c(I)c1 c1(C(=O)OCC)nccnc1NC(=O)CC1CCN(Cc2cc(C)on2)C1 N1(C(c2[nH]cc(CN(C)C)c2)=O)CCCN(C(=O)CCc2cccc(O)n2)CC1 c1(N(C)Cc2cncn2C)ccc(I)cn1 C1(NC(C2(CNC(=O)OC)CCCC2)=O)CC(C)N(C(C2CC(F)(CO)C2)=O)C1 C1(CNC(c2cc(C3CC3)on2)=O)CCC(NC(C2CCOCC2)=O)C1 C1(CNC(C(F)OC)=O)CC(O)CN1C(=O)C(C)CCc1ccc(F)cc1 c1(C(=O)NC(C2CCN(C(c3cnco3)=O)CC2)C)ccc2c(c1)C(=O)NC2 C(=O)(C1=Cc2ccccc2C1O)NCC(C)N(C)C(c1coc(Cl)c1)=O N1(C(C(=O)NC)=O)CCC2CCN(C(c3cc(C(C)(C)C)[nH]c3C)=O)C2C1 N1(C(COCC#C)=O)CCC(F)(C(=O)NCC2CC(O)C23CCC3)CC1 CCC(C(=O)NCC(C)CC1(C(=O)O)CCC1)c1ccccc1 C1(Nc2ncnc(NC(c3cccc(C)n3)CC)c2C)CC2(CCCOC2)C1 CC(C)C(C)C(C)CC(=O)NC1(CNC(=O)CC2CC(C)OC2C)CCC1 c1(C(=O)NCCNC(c2ccc3ccoc3c2)=O)nc2ncc(Br)cn2n1 c1(OCCC)cncc(C(=O)NC(C2CN(C(C3CC3C)=O)C2)C)c1 Cc1ccc(N(C2C3OCC(C3)CNC2=O)C)nc1.C1(CN)CCOCC1 c1(N2CC(C)CC(NC(C)=O)C2)cc(=NC2COC(C)(C)C2)[nH]c(C)n1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1(CNC(C(CC)OC)=O)CCCC1 n1(CCC)nnnc1C(C1CCCOC1)NCCOCCF.OCC n1(CCC)c(COC(C)C(=O)NCCOc2ccc(Cl)cc2)nc2ccccc12 C1(NC(CC2(C)CCC2)=O)CC2CN(C(=O)C(c3cccnc3)O)CC2C1 C1(N(C(=O)C(C)C2CCCC2)CC(C)C)CCN(C(=O)CCn2cnnn2)CC1 C1(CNC(CC(=O)OC)=O)CN(C(c2ncn(C)n2)=O)CC1c1ccccc1 C(C1CCCN1C(C1CC1[N+](=O)[O-])=O)=CC(=O)NCC(C)CO C1(NC(c2nnn(CC)c2C)=O)CCN(C(=O)C(c2ccccc2)O)CC1CO Cc1c(Cl)cnn1CC(=O)NCCN(C(C1CCCN(C(=O)C(C)C)C1)=O)CC C(C(C(=O)NC(c1cnn(C)c1)C)C(C)C)NC(c1cc(CCC)on1)=O C12(NC(Cc3cc(COC)on3)=O)CCC1CN(C(C1(C(F)F)CCCC1)=O)C2 CC(C)CC(C(=O)NCC12CC(NC(c3n[nH]cc3F)=O)(C1)C(C)O2)C(C)C Cn1nnc2c1CCN(C(C1(C)C=CCN1C(=O)C(O)C1CCCC1)=O)C2 C1(NC(C(Cc2ccccc2)N(C)C)=O)CC(F)CN(C(=O)C(F)(F)CO)C1 C1(C#N)(CC(=O)NCC2N(C(c3cn(CC)nc3)=O)CCC2CC)CCCCC1 c1(C(=O)NCC(C)(C)NC(CCC(=C)Cl)=O)c(F)cc(OC)c(F)c1F N1(C(C(C)OC)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)COc1cn[nH]c1 c1(C(=O)NCC2N(C(CCC#CC)=O)CCC2C)cc(OC)c2nn(C)cc2c1 Cc1ccccc1C(C)CC(=O)NCC(F)CNC(=O)C(C)(C)NS(C)(=O)=O C=CCC(C)(CC)C(=O)NC1CCN(C(=O)CC(C=C)CCC)C1CC C1(=O)CC(O)CN1.c1(-n2cc(C3C(C(=O)OCC)C3(C)C)nn2)ccccc1C c1(OCC)ncc(F)c(=NC(=O)C2CC2Nc2ncc(SC)cn2)[nH]1 C(CC(CC)C(=O)NC1CCOCC1C(=O)NC1COCC(C)(C)C1)=CC C(=O)(CC(C)(C)C1CCCCC1)NC1C(NC(C(CC)N(C)C)=O)C1.C1(C)CC1 CN1C(=O)CC(NC(C2CN(C)CCN2C(C2CCC(C)(C)OC2)=O)=O)C1=O Cc1cc2nc(NC(C)CCNC(=O)C(O)Cc3cnc[nH]3)cc(=O)n2o1 c1(NCC(CC)CCO)ncc(S(=O)(=O)N2CCC(C)(C)C2)cc1Cl Cc1nc(C=CC(=O)N(CCCOCCNC(=O)C(C)N(C)C)C)cs1 c1(N(CCCNC(c2cc(C(F)(F)F)ccn2)=O)C(C)C)ccnc(C#N)n1 C1(N(C(C=C(CCC)C)=O)C)CCC(NC(c2nccn2CC)=O)C1 N1(C(c2scc(C)c2)=O)CCC(CNC(=O)CCC(=O)N2CCOCC2)C12CC2 c1(C(N2CCC(C)C(NC(c3ccc[nH]3)=O)C2)=O)cc2nnn(C)c2s1 c1(C(=O)NC2CC(C)(NC(CCC=C)=O)C2)ccc(Cl)c(S(C)(=O)=O)c1 C1(C2(C(N(CC(CN(C(C(c3ccnn3C)C)=O)C)O)C)=O)CC2)CCCCO1 C=CC1OCCC1C(=O)NC1(CF)CCN(C(=O)CCc2cnn(C)n2)C1 c1(C(N2CCCC(NC(CSCC=C)=O)C2C)=O)csc(S(C)(=O)=O)c1 C(=O)(C(CCF)NC(=O)CS(=O)(=O)NC)N(CC)Cc1ccoc1 N1(C(c2ccon2)=O)CCCCC1C1CCCN1c1ncc(O)cn1 c1(C(=O)NCC2(NC(c3c(OC)cccc3)=O)CCOC2)c[nH]c(=N)nc1C N1(c2ncc(CC)c(C)c2)CC2CCC(NC(c3ncoc3CC)=O)CC2C1 C1(CCC(=O)NCCC(C)N(C)C(C2CCCC2F)=O)CCCC(=O)N1 C#CCCC(C(=O)NC(c1cc[nH]n1)C)NC(=O)C(C)C1(O)CCC1 c1(C(C)C(=O)Nc2ccc(OCC(C)O)cc2)c[nH]c2ccccc12 C=C(Cl)CC(C(=O)Nc1cc(O)ccc1F)NC(c1cccnn1)=O N1(C(C2CCC(=O)C2)=O)CCC2(CC(C(=O)NCc3ncsn3)C2)C1 c1(NC(N2CCC(CC3(O)CCC3)C2)=O)nc2cc(C(F)(F)F)ccc2o1 n1(CC)ncc(Br)c1C(N1CC(CNC(C2C3CC4C(C3)C24)=O)C(O)C1)=O c1(C(=O)OC)cccnc1N1CCC(C(C)NC(c2cc(C(N)=O)[nH]n2)=O)C1 Cc1cc(N2CCCC(C(C)NC(=O)C(C3CC(F)(F)C3)O)C2)ncc1[N+](=O)[O-] Cc1cccc(-n2nc(C(=O)N(C(C)CN(C(=O)CC3CC3)C)C)cc2C)c1 C(CC(O)C(=O)NC1CCCC12CC2)NC(COCC#C)=O CC1CC(NC(C2CCC(C)(C)C2)=O)CCN1c1ccc(C#N)nc1 C1(NC(=O)NCCN(CC)CC)CCCC1C(=O)OC.c1(C)ccccc1 c1(N2CCC(CNC(Cc3ccn(C)n3)=O)C23CCC3)cccc(F)c1[N+](=O)[O-] CCC(C)C(C(=O)N1C(C(N2CCCC(O)CC2)=O)CCC12CC2)N(C)C C(CCCCCN(C(=O)Cn1nnnc1C)C)NC(c1c(C)scn1)=O C#Cc1ccc(C(=O)NC2CCN(C(c3c(Cl)ccc(C)c3F)=O)C2)cc1F N1(C(COCCC=C)=O)CC2(CCN(C(c3ccc(C(C)C)c(Cl)c3)=O)C2)C1 c1(C(=O)NCCN(C(CC=C(C)C)=O)C)nc(C)c(C)cc1N CC1(C(=O)NCC2CCN2C(=O)CC=C(Cl)Cl)COc2ccccc2O1 c1(C(N(CC(C)NC(c2ncncc2Br)=O)C)=O)ccc2c(c1)CCC2 CON(C)C(=O)C1(NC(=O)C(F)CC2CC2NC(=O)CC2CCC(=O)C2)CC1 C1(n2cc(NC(c3cc(CC)on3)=O)nn2)CCN(c2ncncc2Br)CC1C C1(C(=O)NC2(CC=C)CN(C(=O)Cc3cc(C(F)(F)F)n[nH]3)C2)CC=C(C)CC1 C1(C(=O)NCC2N(C(C3(C)CCC(F)(F)C3)=O)CCC2)CCCCCC(=O)C1 C1(N(C)C(c2cc(F)n[nH]2)=O)CCCN(C(c2c[nH]nc2C2CC2)=O)C1 C(=O)(C(C)(C)CCCNC(c1nnsc1N)=O)NCC(C(CC)CC)O c1(OC(C)C(=O)OC)ccc(-n2cc(CN(C(CC(=O)OCC)=O)C)nn2)cc1 N1(C(c2[nH]cc(COC)c2)=O)CCN(C(c2ccc([N+](=O)[O-])cc2)=O)C2CCC12 CC1=C(C)CC(C(N2CC(O)CCC2C(=O)NCc2ccc(C#N)s2)=O)CC1 C1(C(N(C2CCN(C(c3c(C)n(CCO)cc3)=O)C2)C)=O)Cc2nncn2C1 C(C)(C(CC(=O)NCc1ccc(C)c(O)c1)NC(C1CC2CCC2C1)=O)OC c1(C(=O)NC(C(C)NC(C2CCCC2)=O)C)cn(CC2CCOC2)nn1 C1(CNC(CCC=C)=O)CCCCN(C(c2cc(CC)ccc2C)=O)CC1 c1(OC)cccc(C(N2CCN(C)CC2CNC(=O)CC2(CC3CC3)CC2)=O)c1C c1(OC)cc(C(=O)NC2CC2CNC(=O)Cc2ccccc2O)cnc1OC C(=O)(CCC(C)(F)F)NC(CNC(CC(C)c1cccnc1)=O)(C)C1CCCC1 C1(C(=O)OCC)OCCN2CC1C2=O.C(=O)(C(S)C(C)C)N(CC(=O)OC)CC c1(N(C)C)cc(F)c(S(=O)(=O)NC(C2CCCC2)C2CCC2)cc1Br CCC(CCC(=O)NCCCC(C)(C)O)NC(C1C2CCC(C2)C1C)=O C1(C)(C(C)C)CCN(C(=O)CCCCNC(=O)C(C)(C)C(N)=O)CC1 C(=O)(CC(O)CCCCC)N1CCC(NC(c2ccc(C#C)cc2OC)=O)C1C c1(N(C)CC2CCC(F)(F)C2)nc2ccccc2nc1N(C)CCc1nccs1 c1(C(N)=O)nc(C(=O)NCC=CCOCC2CC2)cs1.C12(CCOC1)C(=O)N2 N1(C(c2ccc(CC(=O)OCC)cc2)N2CCN(C)CC2)C(=O)NC(CC)C1=O N1(C(C2C(=C)CC2)=O)CCN(C(c2cc(C)cc(C)n2)=O)C2CCC12 N1(C(C(c2c(C)noc2C)(C)C)=O)CC(NC(C2CC2(C)Br)=O)CC2(CCC2)C1 c1(C(=O)NCC(O)CNC(=O)C(F)(F)C2CCCC2)cc2ccccc2[nH]1 c1(C(N2CC(N(C(CCNC(C)=O)=O)C)C2)=O)nc2sc(C)cn2c1C C1(C(C(=O)N(C)C)N(C(C)C)C2CC2)CC2(CCN(CC3CCCO3)CC2)C1 C1(NC(=O)C(F)F)CCCC12CCN(C(C1(CO)CCC1)=O)C2 c1(C(=O)NCC(CNC(C(C(=C)Cl)(C)C)=O)F)cn2cccc(Br)c2n1 N1(C(C2N(C(C)=O)CCC2)=O)CCOC2(CCN(C(C3(CC(C)C)CC3)=O)C2)C1 O=C(C1=CCC(NC(c2csnn2)=O)C1)NCCCc1ncccn1 N1(CC(=O)NCC2CCN(C(c3scc(OC)c3)=O)C2)CCCNC1=O C=C(C)CN=C(NCC1CCN(S(C)(=O)=O)C1)N(C)Cc1cccc(O)c1C c1(CNC(c2ccc(-c3ccc(NC)nc3)cc2)CC)cc(C(=O)O)ccc1F C1(NC(C=CS(C)=O)=O)CCCC12CN(C(C1CC1c1cccc(Cl)c1F)=O)C2 N=c1ncn(CC(=O)NC2CN(C(=O)CSc3cccnc3)C2)[nH]1 Cc1cc(CC(=O)NCc2ccc(C(=O)NCc3nncn3C3CC3)o2)on1 c1(C(=O)NCC2N(C(=O)CNC=O)CCC(C)C2)ccc(S(N)(=O)=O)c(Cl)c1 C12(OC)CCC(C(N3CCC(C(F)(F)F)C(NC(C)=O)C3)=O)(CC1)C2 N1(C(c2cncc(C(N)=O)c2)=O)CC2CC(NC(=O)CSc3cccs3)C1C2 c1(C(=O)OC)cc(S(=O)(=O)NC(C(F)(F)F)c2ccc(C)o2)cs1 C1(CC(C)C)CC(O)CN1C(C1CS(=O)(=O)C1)C(=O)NCCC1(C)CC1 Cc1ncc(C=CC(=O)N(CCCNC(c2ccn(C(C)C)n2)=O)C2CC2)s1 N1(C(=O)NC(COC)C)CCOC(c2ccc(OC)o2)C1 c1(CCF)nc(C(n2cccn2)C2(CC3CCC3)CC2)n(C2CC2)n1 CC1CCC(CCNC(=O)CC2CCN(C(=O)CC3CCCCO3)CC2)C1(C)C c1(CNC(=O)NC2(C)C(C)C2)cc(C#N)cc2ccccc12 C(C)(CSC)(C(=O)NCC1CCCN(C(=O)C(c2ccccc2)N(C)C)C1)OC C1(NC(c2c(C)n(CCO)nc2)=O)CC2CCC1N(C(=O)CCC1CC1(F)F)C2 c1(C(N2CC(CC(CNC(CC=CC)=O)(C)C)C2)=O)cncc2c1CCCC2 C1(NCCNC(CC2(CC)CCC2)=O)CCCN(C(C2CC=CCC2)=O)CC1 c1(OC)cccc(SC)c1.C1(CNC(=O)OCC)CCCCN1C(C)CC(=O)N c1(C(N2C(C)CCC(NC(CCC(C)C)=O)C2)=O)ccc(Cl)c2c1OCCO2 N1(C(c2c(C)cc(F)s2)=O)CCC2(CC1)CCN(C(C1C3CCCOC13)=O)C2 Cc1ccnn1CC(N1CCCC1CC(=O)NC(C)C(=O)NC(C)(C)C)=O S(=O)(=O)(c1cccc(C2CC2)c1)NC(c1ccc(CCCN)o1)=O CC(CC(=O)N1CC2(CCN(C(c3ccc4nc[nH]c4n3)=O)C2)C1)C(F)(F)F N1(C(=O)CC2CC2)CCN(C(=O)C(O)C2CCC2)C(CC2CC2)C1 CC1CCC(NC(=O)Cn2ccc([N+](=O)[O-])n2)CN1Cc1ccc(F)c(F)c1 c1(N(C(c2ccc(C(F)(F)F)c(Br)c2)=O)CC)cc(OC)c(C2CC2)nn1 c1(C(C)N(C(CCC)(C)c2nnnn2CCC2CC2)CC2CC2)c(C)noc1C C1(C(N(CC(C)NC(C2(CCF)CCOCC2)=O)C)=O)CCc2nnc(O)n2C1 C=CCC(C)(C)C(=O)NC1CCC1NC(c1ncc(C)cc1C)=O NS(=O)(=O)CCCC(=O)N1CC(C2(CNC(C34CCN(CC3)C4)=O)CC2)C1 CC1CCN(C(=O)Cc2ccnc(Cl)c2F)CCN1C(=O)CC1(C)CC1(F)Cl C=CC(CC)CC(=O)NC1CCN(C(=O)CSc2ccc(C(N)=O)cn2)C1(C)C N1(C(=O)Nc2n(C)cnc2-c2ccccc2)CCCC2CNC(=O)C12 C(CC(=O)N1CCC(C(N2CCOC(CO)C2)=O)O1)=CC=C.C1CC1 c1(C(N(CC(C)NC(c2cc(F)n[nH]2)=O)C)=O)ccc(C(F)(F)F)cn1 N1(C(C2CCC(=O)N2)=O)CCOC(CNCc2ccncc2O)C1 c1(C(N(CCCNC(c2ccoc2)=O)CC)=O)ccc2ccccc2c1F c1(C(=O)NC2CC(C)CN(C(C3CCCS3)=O)C2)cc2ccccc2cn1 n1(CC)ccc(NC(C2CCCOC2)c2nnnn2CC2CC(n3cccn3)C2)n1 C1(N(C)C(C2CCC(n3cc(Cc4ccncc4)nn3)C2)=O)CCCC1C#N N1(C(C=C(C)CNC(=O)C2=CCCC2)=O)CCOC(C)(C)C1C n1(Cc2nc(-c3ccc(C(=O)Nc4n(CC)ccn4)o3)sc2)ccc([N+](=O)[O-])n1 N1(C(c2n[nH]c(CC)c2Br)=O)CC(NC(=O)C(C)CO)CC2(CCC2)C1 Cc1cc(C(N2CCN(CCC3CCCO3)CC2)=O)nc(C(C)C)n1 N1(C(CC2C(C)(C)OCC2)=O)CCC2(CCN(C(c3coc4c3CCCC4)=O)C2)C1 c1(C(N2CC(C)(CNC(C(COCC)C)=O)OCC2)=O)ccc2[nH]ccc2c1F CC(C)C(C(=O)NCC(O)CNC(C1CCCC1C(F)F)=O)NC(N)=O CN1CCC(C(=O)NC2(C(C)(F)F)CC2)(NC(C2OCCC2(C)C)=O)C1 C1(Cc2n(C)cnc2)OC2(C)CC1(C(=O)NCC(=O)O)C2 CCC(F)C(=O)NC1CC(F)(CNC(c2cn[nH]c2)=O)C1 c1(OC)ccc(O)c(NC(c2cc(OCc3ccccc3)cc(Br)c2)=O)c1 Cc1cc(C(=O)NC2CCC(NC(c3nocc3C(C)(C)C)=O)CC2)nc(O)c1 C(C1CN(C(=O)CN(C(=O)COC)C)CC1C(=O)NC1CC(Cl)(Cl)C1)=CC c1(N(CC(C(C)C)C)C)ncc(S(=O)(=O)NCC2(C)CSC2)cc1Cl C1(NC(C(C)SCCCC)=O)CC=C(C(=O)NCc2nc(C)sc2C)C1 N1(C(C2CN(CC)C(=O)C2)=O)CCCC(C2CN(C(=O)COCC3CC3)C2)C1 c1(C(N2CC(CNC(CC(C)F)=O)C3(C2)CC3)=O)nc2ncccn2n1 CCCCC(O)C(=O)N(C)CC1CN(C(c2ccc(C#N)o2)=O)CCO1 C(C1=NOC2CCCCC12)n1cc(CN(C2CCCC2)C)nn1 C12(C(N(C3CCN(C(=O)CC4(CSC)CC4)C3)CCC)=O)CCC(C)(CC1)OC2 C1(NC(=O)Cn2ccnn2)CCOC(C(N2CCC(CO)C2)=O)C1 C(=O)(C1CCc2cccnc21)N1CCN(C)CC1CNC(c1cc(C#N)c[nH]1)=O CC(C)C(C#N)C(=O)N(CCN(C(=O)Cc1cccc(C(N)=O)c1)C)CC1CC1 Cc1cncc(CNC2CCCC2NC(C2CC3(CCC3)C2)=O)c1 c1(C(N(C(CC)CNC(C2CC23CCC3)=O)C)=O)cc2cccnn2c1 N1C(=NCCCF)NCC2(CCOCC2)NC(=O)C1.c1(NS(C)(=O)=O)cccc(Cl)c1 C(=O)(C1=CC2CCC1C2)NC1CC2CN(C(c3cc(C(CC)CC)no3)=O)C1C2 c1(C(=O)NC(c2onc(C)n2)=O)ccc(CC2CC3CNCC23)cc1 c1(C(=O)OC)cccc(C(=O)NC(CO)C(C)NC(c2ncoc2C)=O)c1 c1(C(=O)NCC(N(C(C(C(C)O)N(C)C)=O)C)C2CC2)cnc2[nH]cnc2c1 c1(CC(=O)NCC(CNC(c2n(CC)ccc2)=O)C)cccc(-c2ccco2)c1 C(=O)(C1CCOc2ccccc21)NCC1C(C)CN(C(C2(C)COC2)=O)CC1 c1(C(N(CCC=C)CC(F)F)=O)cc(CCN)on1.C(=O)(C=CC(F)F)NCC=C Cc1cc(C2(NC(C3(CNC4CCCN4CC(F)(F)F)CCC3)=O)CC2)on1 C#Cc1cncc(C(=O)NCc2cc(O)cc(F)c2)c1.C12(CCCC1C)C(=O)N2 N1(C(C(CCC)CC(C)C)=O)CC(C2CCCN(C(C3CC=CCO3)=O)C2)C1 C12(C(N3C(CNC(CC)=O)CCC3)=O)CCCC1CCN2C(C1CC=CC1)=O C1(C(=O)NCC(CC)NC(=O)COC2CCC2)CC(=O)c2cc(Cl)ccc2O1 c1(SCC(=O)NC(C(C)NC(C(C)NC(=O)NC)=O)(C)C)ccnc(O)c1 c1(C(N2CC3C(CNC(CCCCC=C)=O)(C3)C2)=O)ccc(F)c2cccnc12 C(CC(CC)C(=O)N(C)CCNC(c1ccsc1COC)=O)=CC c1(C(N2CCC(NC(=O)C(=O)c3ccco3)C(F)C2)=O)cc(Br)cc2ccccc12 N1(C(c2cc(C)cc(C)c2)C(=O)NC2COC2)CC2CCN(C)CC(C2)C1 C(=O)(CCC(CF)CF)N(C1CCN(C(=O)C(C)C(C)(F)F)C1)CCC CN1CCN(C(=O)CCc2ncc[nH]2)C(CNC(C2(C)CCCO2)=O)C1 C1(CNC(CC(c2ccc(OC)cc2)C)=O)CN(C(=O)C2=CCC2)CC(C)(C)O1 C1(CC(=O)OCC)CCCN1N1CC(C)(C)OCC1C c1(C(N(CC(C)NC(=O)CC(C)(C)C(F)F)C)=O)ncn2cc(Cl)ccc12 C=CCC(C)C(=O)N1CCCC1C1(O)CN(C(=O)CCc2ccc(OC)cc2)C1 C1CN=C2C=C(C)N=C(N2)SCCO1.c1(C(=O)OC)ncn2c1CCCCC2 C1(C)(C(=O)NCCCN(C(C2C(C=C)C2)=O)C(C)C)CCNC1=O C(N=c1cc(N2CCC(CF)C2)nc[nH]1)c1ccnc(C(C)(C)C)n1 c1(OCC)cc(C(N2CCCC2CNC(C2CC2c2ccccn2)=O)=O)ccn1 C1(CNC(c2c(C)ocn2)=O)CN(C(c2nccc(Cl)c2Cl)=O)C2(CCC2)C1 N1(C(c2nc(COC)sc2)=O)CCOCC1CNC(=O)CCc1cccs1 c1(C(=O)NCCc2cscn2)cc(CNC(C2CC2c2cccnc2)=O)ccn1 C12(NC(CCN(C)CCO)=O)CCOCC1CN(C(=O)Cc1cn(C)nn1)C2 c1(C(N(CCC(=O)NCC(C)C(F)F)C)=O)n[nH]c2c1CCC2 C1(CNC(C(c2c(F)cccc2F)C)=O)CCCCN(C(=O)C=CC=C(Cl)Cl)C1 C1(NC(Cc2ccc(C)cc2)=O)CCCCN(C(=O)C(=O)NCC(F)F)C1 c1(C(N(C2CCOC2)CCNC(=O)OC(C)(C)C)=O)cncc(Br)c1 C1(C(N2CCCC2C2(C(=O)Nc3cncc(CO)c3)CC2)=O)CCCC2(CC2)C1 c1(C(N(CCCNC(C2CCNC2=O)=O)CC)=O)c(C)ncn(C)c1=O C(CCCC(=O)NC1CCCC1(C)CNC(=O)Cc1cn(C)nc1C)OCC Cc1cn2cc(C(=O)NCC(O)CNC(=O)C(C)S(C)(=O)=O)ccc2n1 C(=O)(C(C(=O)N(CC(C)NC(=O)C(F)(F)c1cscn1)C)C(C)(C)C)OCC N1(C(CS(=O)(=O)NCC)=O)CCC(NC(=O)CCCCCN(C)C)C12CC2 C1(CNC(C(CNC(C(c2cnn(C)c2)C)=O)(C)C)=O)CCOCC1(C)C CCC(CC(=O)N(C)CC1(O)CN(C(c2ccnc(C(N)=O)c2)=O)C1)OC Cc1ncnc(C)c1CC(=O)NC1CC12CC(NC(=O)C=CC(C)C)C2 Cc1ccc(F)c(CNCc2cn(C)nn2)c1 Cc1nc(C)c(C(=O)NCCC(C)CCNC(=O)Cc2cncc(Br)c2)o1 c1(C(C)(C)C)cc2c(Nc3ccccc3NC(C3(F)CCNC3)=O)ncnc2s1 c1(C(N2CCC(C)(NC(c3c(CC)sc(=N)[nH]3)=O)C2)=O)c(Cl)ccc(Cl)c1O C1(CC(=O)N(C(c2ccccc2)CO)C)C(C)(C)C1(C)C c1(C(=O)NCC(CO)NC(C(CC(C)C)(F)F)=O)cnc(O)c2ccsc12 C1(C(C(=O)NC2CC(CC)C2)(C)C)CCCN(C(=O)CC(Cl)Cl)C1 C1(NC(C(CC)F)=O)CC2(CCN(C(=O)CCN3C(=O)CCC3=O)CC2)C1 Cn1ncc2ccnc(C(N3CCC(C4CC4)(CNC(C4CCSC4)=O)C3)=O)c12 c1(C(=O)NC(CNC(C=C(COC)C)=O)C2CCC2)cnc2ccccn2c1=O O=C(C#CC1CCCCC1)N1CC2CC1CN2C(c1c(Cl)ccc(O)c1Cl)=O CCC(C)C(=O)N(CCOC)CC.C12(C)CC(C1)NC2=O.C(=O)(NC)O C1(C(N(CCCOCCN(C(CCC(=C)C)=O)C)C)=O)CCC(=O)N(C(C)C)C1 N1(C(C(=O)N(C)C)=O)CCC(CCNC(C2CCCC(F)(F)C2)=O)C(F)(F)C1 c1(OC)cncc(C(N2CCC(C3CCCCN3C(c3cc(CO)on3)=O)C2)=O)c1 C12(C)CC(CN1C(=O)CN(C)C1CC1)NC2=O.c1(COC)ccc(O)c(F)c1 c1(C(=O)NCCn2cc(C(=O)NC(C3CCC3)CC)nn2)cc(C)n(C)n1 c1(OC)cc(C(=O)NC2CN(C(C3CC(C(F)(F)F)C3)=O)CCC2O)ccc1O c1(SCNC(C2C3CC(C)N3N2C)=O)ccc(Br)cc1.C1(CC)CCCC1 c1(C(=O)OC)ccc(C(F)(F)F)nc1NC1CCCCC1c1ccccc1 CCC(C(=O)N1CCC(C)CC1COC)C(C)(C)CC.O1C(=O)C2(CC2)C1 CCC(C)CC(=O)C(=O)NCC(C(C)(C)C)NC(=O)Cc1cn(CC)nn1 c1(OCC)ccc(C(=O)NC(CNC(C2(CC(F)(F)F)CC2)=O)CO)cn1 CCCC(C#N)C(=O)N(C(C)CC(=O)NCCn1cnnc1C)C c1(C(N2CCN(C(C(CC)OC)=O)CC2CC)=O)nn(C)cc1[N+](=O)[O-] c1(OCC)cc(Br)cc(C(N2CCCCC(NC(C3CN(C)C3)=O)C2)=O)c1O C12(NC(c3ccc(CC)cc3Cl)=O)CCCN(C(=O)C(C)(C)C)CC1C2 C1(CNC(C(c2nc(C)sc2)=O)=O)(NC(C2CCC2)=O)CCC(C)(C)CC1 O=C(CCCC1CC1)NCC1CC1NC(c1ccnn1CC(F)(F)F)=O c1(C(N2CCN(C(C3(CC)CC3)=O)CC2CC(F)F)=O)ccc2c(c1)C(C)CO2 N12CCC(C3CCCC3C1=O)CC2.c1(CSC(C)(C)C)nc(O)n[nH]1 C=CCC(C)(C)CC(=O)N(C1CCN(C(=O)CCC(C)(F)F)C1)CC c1(C(=O)NCC2N(C(C(C)Cc3ccncc3)=O)CCCC2)ccnc(F)c1F N1(CCCC)C2CCC1CN(C(=O)NCC(c1ccncc1)OC)C2 c1(CN2CCC(C(=O)N=c3cccn[nH]3)CC2)ccc(F)c2ncccc12 c1(CC(N2C(CC(=O)NC3CCC(F)(F)C3)COCC2)=O)c(F)cccc1F N1(C(c2c(CC)cc[nH]2)=O)CCC(C)(C)C1C(N1CC(CNC(=O)OC)C1)=O n1(CC(=O)NCC2CC(NC(COC)=O)C2(C)C)ccc2cc(OC)ccc12 Cc1cc(-n2cc(CC3CN(C(C)C(c4ccc(F)cc4)O)C3)nn2)cnc1Cl Cn1cnc(C(N2CCC23CN(C(=O)CCC2CCC4(CC4)CO2)C3)=O)cc1=O C1(NC(c2c(CC)nco2)=O)CC(NC(=O)CC2NC(=O)NC2=O)CC1O C#CC(C)(C)C(=O)N1CCC(C2OCCC2NC(=O)COCCCOCC)CC1 c1(CN2C(C(=O)Nc3cccnc3Cl)CC(F)C2)cc2cnccc2[nH]1 c1(C(NOC(C(=O)OC)C)=O)ccn(CCNC(=O)C=C2CCCCC2)c1 C=Cn1nccc1C(=O)N(CC(C)(C)CNC(C1CN(c2ccccc2)C1)=O)C c1(C(=O)NC2CCCN(C(CCOC(C)C)=O)C2)[nH]c2ccccc2c1Cl c1(Nc2cnc(C(C)(C)C)cn2)cccc(C(=O)Nc2c(C(=O)OC)scc2)n1 c1(C(=O)NCC2C(C)CN(C(=O)CC3CCC3)CC2)ccc2c(c1)C(=O)OCC2 c1(OC)cnnc(C(=O)NC2COCC2CNC(=O)C(=C2CCCCC2)F)c1 CC1CN(C(=O)C2=CSCS2)CC2(CCN(C(=O)C(C)(C)C(N)=O)C2)O1 Cc1cc(F)ccc1CC(=O)NC1C2CC1N(C(=O)C(F)(F)C(O)C1CC1)C2 c1(C(N2CCC(O)(CNC(c3c(C)occ3)=O)C2)=O)cc(C(F)(F)F)ncc1N CP(C)(=O)c1cccc(C(=O)NCC2CN(C(C3CCC(N=[N+]=[N-])C3)=O)C2)c1 C1(CC)CN(C)CCCN1C(c1ccc(CNC(=O)C(=O)C(C)(C)C)nc1)=O N1(C(c2c(C)cno2)=O)CCC2(CC1)CC(C)N(C(=O)CCN1CCC1)C2 c1(OCC(C2CC2)NC(=O)C=CCN2CCCC2CC(=O)C=CCl)ccccc1 C(c1ccc[nH]1)=CC(=O)NCC1CCN(C(=O)Cc2ccc(C(=O)OC)s2)C1 c1(C(=O)NCC(C(C)C)NC(=O)C=CC=C(Cl)Cl)ccc2c(c1)SCC(=O)N2 N1(C(COCCCC(C)C)=O)CCCC2(CCCN2C(C2CSCCS2)=O)C1 c1(C(N2CC3C(CNC(CCC=C=C)=O)(C3)C2)=O)ccc(N)cc1Cl C1(CNC(C=CCC)=O)CCCCN(C(c2c[n+]([O-])c(C)cn2)=O)C1 N1(C(c2nc(C)n(C)n2)=O)CC2CC(CNC(=O)C(C)Cc3ccco3)C2C1 Cc1nccnc1C(=O)NC(C)C(C)NC(c1cnccc1Cl)=O c1(C(=O)NC(CN(C(C2CC(C(F)(F)F)C2)=O)CC)C)cc(C)c(C)cc1N C1(C(=O)NCC2(CNC(C3C(C)(CC)C3)=O)CC2)C2CC3C(C2)C13 C1(NC(C(C)S(C)(=O)=O)=O)CN(C(=O)C2=CCCS2)CC12CCOCC2 C(=O)(CC1=NNC(=O)C1)NCCCC(CCC)NC(C1(C)CC(C)(C)C1)=O N(C(=NCCc1ccccc1)NC(c1ccc(Cl)nc1)C)CC(C)C#N N1(CCOC)CC(CN(C)C(c2ccc(NC(=O)OC(C)(C)C)[nH]2)=O)C2(CC2)C1 c1(C(=O)NCC2CCC(NC(CCOC)=O)CC2)cnn2ccc(O)nc12 c1(C(=O)NC2CCN(C(=O)CSC3CCCCO3)C2)ccc2c(c1)C=CCC2 CC1CC(C(F)(F)F)CN1C(=O)Nc1nccnc1-c1ccc(OCF)cc1 Cc1cc(C(=O)NC2CN(C(=O)C(c3ccccc3)=O)CC2(C)C)c(F)cc1F C#Cc1ccc(C(N2CC(CC(C)NC(=O)CC(=O)NCC)C2)=O)cn1 C1(C)(CC(=O)NCC(COCC)O)CCN(C(c2c[nH]nc2C)=O)C1 c1(C(N2C(CN(C(C(C=CCCC)O)=O)C)CCCC2)=O)ccc(F)cc1C CCCC(C)CC(=O)N1CCOC(C(=O)NCC2CNC(=O)CO2)CC1 N1(C(Cc2cnc(C)o2)=O)CCC2(C1)CN(C(=O)CCCN1CCCC1)CCO2 C(C(=O)NCCC1(NC(c2cnn[nH]2)=O)CCC1)(C(C)(C)C)SC N1(C(C2CCCN(C(=O)OCC)C2)=O)CCC2(CCC2NC(=O)CCC)CC1 c1(NC(C2CC(=C)CN2C(c2ccc(C3CC3)cc2C)=O)=O)cccc(C)c1O C#Cc1cncc(NC(c2cnnn2C=C)c2nnnn2-c2ccc(F)cc2C)c1 Cn1cc(S(=O)(=O)NCC2CCN(C3CCCCCC3)CC2)c(O)nc1=O C1(CNC(C2N(C)C(=O)NC2)=O)CCCCN(C(C2(C#N)CC3(CC3)C2)=O)C1 Cc1ccc2[nH]cc(CC(=O)NCC3CC(F)CN(C(=O)CC(C)F)C3)c2c1 C1(OCC(=O)OC)COC2CN(C(=O)C(=O)NC(C)(C)CCCOC)CC12 C1(CSC)CCN(C(=O)Cn2cnc(C(F)(F)F)n2)CC1 C1(C(=O)NCC(CC)NC(=O)C(N2CCN(C)CC2)C)CC2(C1)CC(C)C2 N1(C(c2c(C)oc(CO)c2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC(O)C1 C1(COC)CN(C(=O)CC2(COC)CC2)CCN1C(c1cc(O)nn1C)=O C(C(C)C(=O)N1CCCC1CN(C(c1cnc[nH]1)=O)Cc1scnc1C)OC N1(C(CNC(=N)N)=O)CCC2(CC1)COC(C(=O)N(c1nccc(Br)c1Cl)CC)C2 c1(C(N2CC(O)(C(C)NC(C3CCCCNC3=O)=O)C2)=O)cc(F)c(F)cc1N N1(C(C2=CCC(NC(CCCC(C)C)=O)C2)=O)CC(C)c2ncccc21 C#CC1(C(=O)NCCC(C)(C)CNC(c2cscc2CC)=O)CCCC1 c1(C(N2CC(NC(CC(C)C)=O)C3(C2)CC3)=O)cc(F)c(F)c(Cl)c1F N1(C(C=CCOC)=O)CCCC2(CCC(NC(=O)CNC(=O)CC(F)(F)F)C2)C1 C12(C(=O)OCc3onc(COCC)n3)CCOC1CC(=O)NC2 c1(C(N(C2CN(C(C3C(=C)C3)=O)CC2(C)C)C)=O)cc2c(cc1Cl)OCO2 Cc1nc(C(=O)NC(c2nocc2C(N2CC(F)(F)C2)=O)C)ccc1C#N C(=O)(C(C(C)C)NC=O)N(CC(=O)N(C(CC)C)C)CC1CC1 Cc1cc(N)ccc1C(=O)NC1CCC(NC(C23CSC(C2)C3)=O)CC1 N1(C(C2CCC(C(C)C)CC2)=O)CC2CC1CN(C(C13CCC(F)C1CC3)=O)C2 Cc1nc(NC(c2cn(C)nc2CC2CCCNC2)=O)c(Br)nc1Br C1(CN(C)C)C(=O)OC2CC(C2)C(=O)N1.c1(CCNCC)cc[nH]n1 C(CC(C)(C)CNC(=O)CCN1C(=O)CCC1=O)NC(C1(CC=C)CCCC1)=O c1(N(C)CC)nc(=NC2CCCN(C)C2C)[nH]c2cc[nH]c12 C#Cc1cnc[nH]1.N12CC(C1)N(CCOC)CCNC(=O)C1C(C1)C2=O.C1C(=O)O1 C1(C)(CNC(CC2CCN(C(c3cc(C)no3)=O)CC2)=O)CC2(CCC2)C1 C1(NC(c2c(C)nn(CC)c2C)=O)CN(C(C2CCCOC2C)=O)CC2(CC2)C1 C1(CCCC)(C(=O)NCCOC(C)(C)CNC(=O)CC2CCSCC2)CCCC1 C1(OC)CC(CC(=O)NC(C)CN(C)C(C23CC(CCO2)C3)=O)C1(C)C N1(C(C(=O)NC(CN(C(c2c(C)c(O)ccc2)=O)C)C)C)CCc2ccccc21 Cc1nccc(C(N2CCC3(CC3C(=O)NCC3CCC(=O)O3)C2)=O)c1C C1(CC)CNC(=O)CN1C(=O)CC1C(NC(c2ccc(F)c(O)c2)=O)CC1O c1(C(N2CCN(C(c3c(OC)cccc3)=O)CC2C)=O)csc2c(O)ccnc12 C1(NC(CNC(C2C(C)C2)=O)=O)CN(C(=O)Cn2cnnn2)CCC12CCC2 c1(CC)cc(C(=O)N(C(C)C(=O)NCC(=O)N(C)O)C2CC2)nn1C C(=O)(CCN(OC)C(=O)c1cccc(NC(c2scnc2C)=O)n1)OC S(=O)(=O)(c1cc(Br)ccc1Cl)N(S(c1cn(CC)nc1)(=O)=O)C1CC2CNCC2C1 c1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)cc(O)nc2cnccc12 c1(C(=O)OC)cc(Cl)ncc1NC(C1CC12CCN(Cc1ccc(CBr)cc1)C2)=O C1(CNC(C2(SCC)CC2)=O)CCN(C(=O)C2=NOC(C)C2C)CC1(F)F N1(C(c2nc(C(C)C)sc2)=O)CCC(N(C(=O)Cc2ccsc2)C)CC1 Cc1onc(C(N2CC3(CCC3)CC2CNC(=O)C(O)C(F)F)=O)c1[N+](=O)[O-] C1(C(=O)NC2C(NC(c3cc(CC)nn3C)=O)C2)COc2ccc(OC)cc2C1 C(=O)(CCCCc1cnc[nH]1)NCCC(C)N(C(=O)C(C)(C)c1ccn(C)n1)C c1(C(=O)NCC2CC3CC3N2C(C2CCCSC2)=O)cc2c(F)cccc2[nH]1 c1(C(C)(C)C)ccc(C(=O)NCCCCCNC(=O)C(F)C2CCOC2)s1 O=C(NNc1nc2ccc(Br)cc2s1)c1ccc(F)cc1.C1(N)CC2CCC(C1)O2 c1(C(N2CCCCC(NC(C3(COC)CCOC3)=O)C2)=O)cc(N)c(Cl)c(O)c1 Cc1cn2[nH]c(=NC3CC(CCNC(C4CSCCS4)=O)C3)sc2n1 C1(NC(=O)Nc2cc(S(=O)(=O)N3CCSCC3)c[nH]2)CCCCC12CCCC2 n1(CCC(=O)NCC2(NC(C3C4(CC4)C34CC4)=O)CCOC2)cccnc1=O c1(C(OC)OC)ncccc1CNC(N1CCCC(c2ncc(C)s2)C1)=O N1(C(C(C=C)O)=O)CCC(C2CCC2)(CNC(c2cc(CC)ccc2O)=O)CC1 Cc1ccc(F)cc1C(N1CCC(C(=O)NCc2ccc(CO)o2)C(O)C1)=O c1(OC)cc(C(=O)NCC(C)(C)CN(C)C(C2(C)CCCN2C)=O)cc(F)c1F N1(C(CN(c2c(CC)cccc2)C)=O)CCCC(CO)C1C=O C(CC)(C(=O)NOCC(N1CCC12CCCSC2)=O)OCC CC1(C)C=C(C(=O)N2CCOC(CCCNC(c3cn(C4CC4)cn3)=O)C2)C1 c1(CC(=O)NC2CCN(C(C3(OC)CC3)=O)CC2C)ccc(C)c2ccccc12 c1(C=O)nnc2ccccc2n1.N12CC(CC(O)C1)Nc1cscc1C2=O.CC=CC CCC(=O)CCC(=O)NCC1CCCC(NC(c2cc(C)n(CC)c2C)=O)C1 Cc1cc(C)c(C(N2CCCC(N(C(=O)Cc3scnc3C)C)C2)=O)c(Cl)n1 c1(OC)cc(C(=O)NC2(CNC(C3C4CC4C4CC34)=O)CCC2)c(F)cn1 c1(OC)ccccc1C(=O)NCC(C)NC(=O)CCOC1CC(C(F)(F)F)C1 N1(C(=O)OC(C)(C)C)CC2(CCC(NCc3cn(C)nc3[N+](=O)[O-])CC2)C1 C12(NC(CNC(CN(C)C)=O)=O)CCCC1N(C(C1CCC(C)(O)CC1)=O)CC2 N1(C(c2cncs2)=O)CC2(CO)CC1(C(N1CC(Cc3ccoc3)C1)=O)C2 CC(C)CC(C(=O)NCC(C(C)C)NC(c1ncnc(O)c1Cl)=O)C(N)=O CS(C)(=O)=Nc1ccccc1C(N1CCN(C(c2cncs2)=O)C(C(F)F)C1)=O C1(C(=O)NC(C(=O)NCCNC(=O)NC)Cc2ccoc2)CC2CCCC2C1 C1(CNC(CN(CCOC)C(C2CC3CC3C2)=O)=O)CCOCC1 C1(NC(c2cnn3cnnc3c2)=O)CC2CN(C(C3CCCC3)=O)CC2C1 n1(CC(=O)NCCN(C(CCOCCC)=O)CC(C)O)nnc(C(C)(C)C)n1 C(C(CC(C)C)C(=O)NC1CCC(C)N(C(c2cccnc2)=O)C1)OC C1(C(=O)NCC2C(C)OCC2)CCCN(C(C2(C(N)=O)CC2)=O)C1 c1(-c2scc(C(C)NCC(c3ccccc3)O)n2)ccc(Cl)cc1 c1(OC)ccc(CC(=O)NCC(C2CC2)NC(c2oncc2C)=O)c(Cl)c1OC N1(C(CCCN(C(=O)OC)C)=O)CCCC(CO)(NC(c2oncc2C)=O)C1 C1(C(N(CCCN(C)C)CCNC(c2cnccc2Cl)=O)=O)CC2(CCOCC2)C1 C1(NC(=O)CN2CCCC2)CC2CC1N(C(c1ncccc1C(F)(F)F)=O)C2 c1(C(=O)NCCN(C(C)C(=O)NCc2ccccc2)C)c(C#N)cnn1C c1(NC(c2cnn(C3CCCCC3)c2)C)cccc([N+](=O)[O-])c1Cl.c1nnnn1C CCC(CCOC)C(=O)NCc1csc(CNC(=O)C(c2ccc(Cl)cc2)O)n1 C(C(C)(C(=O)N(CCCN(C)C)C(C)C)NC(=O)CC(C)n1ccnc1)SC c1(OC)ccc(NC(C2CC23CCN(C(=O)C=Cc2cnn(C)c2)C3)=O)cc1C CCC(C)C(O)C(C)C(=O)N1CCN(C(c2ccn(C)c2C)=O)CC(O)C1 c1(NC(C)=O)cccc(C(N2CCCCC2CNC(C2COC(C)C2)=O)=O)c1 NC1CS(=O)(=O)Cc2ccccc2N1C(=O)Nc1ccsc1 N1(C(c2cc(SCC)on2)=O)CCN(C(C)CNC(c2n[nH]cc2C)=O)CC1 c1(C(=O)NC(CC)CNC(c2ccnn(C)c2=O)=O)cccc2[nH]ccc12 C(C(CC(F)(F)F)NC(=O)CCC(N)=O)NC(COCc1n(C)ccn1)=O C1(NC(C(C)N(C)C)=O)CCC2CN(C(=O)Cc3ccc4n[nH]cc4c3)CC2C1 CC1(C)COc2c(C(=O)OCC3(C)CCCCC3)cccc21 C1(CCC(=O)NCCN(CC(C)O)C(=O)Cn2cnnn2)CCCOC1 C1(NCc2cnn3c2CN(C(=O)OC(C)(C)C)CC3)CCOCC12CCCC2 Cc1nc2ccc(C(=O)NC3COCC3(F)F)cc2[nH]1 c1(C(=O)OC)cnc(Cl)nc1N1CCCOC(CNC(=O)C=CC(=O)N(C)C)C1 c1(C(=O)NCC2CC2(Cl)Cl)cccc2c1OCCN2 CC1CCCCC1N(C(=O)C(c1cccc(Br)n1)(F)F)C Cc1ccc(CN2CC(NC(c3cc(Cl)cc(Br)c3)=O)C(C#N)C2)cc1O C(CC(=O)NC(c1cncnc1)C)(C(C)C)NC(C1(CC#C)CC1)=O CC(C)CC(C)C(=O)N1CCC(NC(c2ccnc(OCC3CCC3)c2)=O)CC1 C(=O)(C1=C(c2ccccc2)SCCO1)NC(C(C)NC(COCC)=O)C c1(C(=O)NCC(CCOCC)NC(c2cnc(OC)s2)=O)cnc(C)nc1 N1(C(c2ccc(NC)cn2)=O)CC(C)CN(C(=O)C(=O)Nc2ncc[nH]2)C(C)C1 C1(NC(C(CC)OCC)=O)CCN(C(=O)CCC(=O)c2ccccc2O)CCC1 C(N=c1nc(O)c2ccc(Cl)cc2[nH]1)C1CN(C(C2=C(C)OCCS2)=O)C1 C12(NC(C3CC(C)C3)=O)CCCCCC1N(C(=O)Cc1ccccc1Cl)CC2 c1(C(C(=O)N(CC(=O)N(CC)CC)C)(C)C)ccc(Cl)cc1.SCC C1(C2CCN(C(=O)CC3CCCSC3)CC2)(NC(c2cnco2)=O)CCC1 c1(S)nc(C)cc(C)n1.C1(C(C)N)CCN(CC2C3CCCC23)C12CC2.C1(=O)CC1=O C(CCC1CC1)(C(=O)NCCCC(F)F)NC(C1C=C(C)CS1)=O c1(C(N2CCC(NC(=O)C(F)OC(F)(F)F)C(O)C2)=O)nccc2c[nH]nc12 c1(NC(=O)Nc2c(CCC)nco2)cnc(C(C)(C)C)nc1 N1(C(=O)Cc2ccno2)CCN(C(=O)COCCc2ccccc2)C(CCO)C1 c1(C(N2CCC(C(C)CNC(C3OCCCO3)=O)CC2)=O)cc2occc2n1C CN1CCCCC(C(=O)NCC2CC2NC(C23CC(C)(C2)OC3(C)C)=O)C1=O C12(CNC(C3CC(C)(NC(=O)CCCN4CCCC4)C3)=O)CCC(C1)C(=O)N2 N1(C(c2cn(CC)nn2)=O)CCOC2(C1)CN(C(C1CCCC13OCCO3)=O)C2 N1(C(C(CCC#C)NC(=O)C(CO)C(F)(F)F)=O)CC2(CC2)CC1C#C C1(C(=O)NCC23CC(CN2C(=O)C(O)CC2CCCC2)C3)CC2CCC1CC2 N1(C(C2C(C)C2)=O)CCC2C(CCN2Cc2ccc(F)c(Br)c2F)C1 N1(C(=O)Nc2sc3c(n2)C(C)CCC3)CC2CCCC2C12CC2 c1(OC)cccc2[nH]c(C(N3CCN(C(c4csnn4)=O)CC(C)(F)C3)=O)cc12 N1(C(CCC(C)(C)O)=O)CC2CCN(C(c3noc4c3COCC4)=O)CCC2C1 c1(C(=O)NCC2OCCC(NC(C(P(C)(C)=O)O)=O)C2)c(Cl)nc2ccccn12 c1(C(C)NC(C=CC(C)NC(=O)COCC(C)(C)C)=O)ccc(O)nc1 C1(C(=O)NC(C2CCN(CC(C)C)CC2)C)CCCC(F)(F)C1 c1(C(=O)NC)ccc(C(=O)NCCC2(O)CN(C(C3CC3(F)Cl)=O)C2)cn1 N1(C(c2cc(C)c(Br)c(C)c2)=O)CC2CCN(C(=O)C(=O)C(C)(C)C)CC2C1 c1(C(=O)NCCN(C(Cc2n(C)nc(C)c2Br)=O)C)onc2ccccc12 N1(C(CC2(NC(C)=O)CC2)=O)CC(O)(c2cn(CC3(F)CCOC3)nn2)C1 C(CCCCC(=O)NCCc1cnn(C)c1C)NC(C(CC)CC)=O c1(OC)cccc(C(N2CCC(C(C)(C)NC(C3CCCCCC3)=O)C2)=O)n1 C(c1ccccc1)=CCC(=O)N(CCn1ccc(N(CC)CC)n1)CC C1(C(=O)NCC(C)(CO)NC(c2cc(F)c[nH]2)=O)CCC(c2ccccc2)CC1 C(=O)(C1=CSCS1)N1CCC(NC(C2CC(=O)N2)=O)C1 c1(CNC(c2cccc(CNC(CC3(OC)CCC3)=O)n2)=O)ccc(O)cc1F N1(C(C)=O)CCC(C)(C)C(NC(=O)CN2CCS(=O)(=O)CC2)C1 c1(NC(C2CCCN2C(c2cnc(S)nc2)=O)=O)ccnc(CO)c1 N1(CCC(C)(C)C)CCC(CNC(=O)C(C)CCCCc2ccccc2)C(C)(C)C1 O=C(NNC(=O)Nc1ccccc1)OCC1CCCN(S(=O)(=O)C(F)F)C1 CC1CC(C(=O)N(C)CCC2CC2)CN(C(=O)CC2(O)CCCCC2)C1 N1(CC(N2C(CN(C(Cc3nnc(C)o3)=O)C)CCC2)=O)C(=O)CN(C)C1=O c1(SC)ccc(NC(C)C(=O)NC2CC2NC(=O)C(=O)Sc2ccc(Cl)cc2)cc1 N1(C(c2c(C)nn(C)c2Cl)=O)CCN(C(C2(OC(C)C)CCC2)=O)CC2(CC2)C1 C12(NC(=O)C=CC=C(Cl)Cl)CCC1CN(C(=O)CSC1CCCCO1)C2 N1(C(c2cn(C)nc2C2CCC2)=O)CCC2CCCC(C1)N2C(C1C=CCC1)=O C(C(F)(F)F)=CC(=O)NCCC1(NC(c2cnn[nH]2)=O)CC1 Cc1ccc(F)c(C(=O)NC2CC(O)CN(C(C3(n4cccn4)CC3)=O)C2)c1O c1(-c2c(C)occ2)nc(C2CC(C)(C)C2)n(CCOCCC(F)(F)F)n1 c1(OC)cccc(C2COC2)c1.C1(=O)C(c2cc[nH]n2)N1 C1(C(=O)NCC2CN(C3CCC3)C2)CCC(O)CN1C(c1cccs1)=O C1(n2cc(CCC(=O)NCc3ncc(Br)s3)nn2)CCCCC1NC(N)=O c1(C(=O)NCC(C(C)C)(C)NC(C2CC(C)(F)C2)=O)cn(C)c(=O)n(C)c1=O C12(CC(=O)N(C)Cc3cccc(F)c3)CCC1CN(C(=O)CC1(O)CCC1)C2 C(=O)(NNc1nc(Cl)ccc1Br)Nc1c(S(C)(=N)=O)nccc1 c1(C(=O)NCCNC(=O)C(O)c2cnc[nH]2)cn(CCSC2CCC2(F)F)nn1 C(=O)(C1CCC(=O)c2cccn21)NC1(CC=C)CN(c2nc3ccccc3o2)C1 c1(C(N2CCC(C(F)F)(CNC(C(C(C)C)SCC)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 C(CCC(C)C(=O)NCCC(O)C(=O)NCCCc1cncnc1)OC c1(NC(C2CC(C)N(C(c3ccnc(Cl)c3O)=O)C2)=O)ccc(O)c(CO)c1 C1(NC(C2(C(N)=O)CC2)=O)CN(C(C2CCC3C(C2)C3(F)F)=O)C2(CCC2)C1 CC(C)C(C#N)C(=O)N1CCCC(C(=O)NCCC(=O)N(C)C)C1C c1(C(=O)OC)cc(C(N2CC=CC2CNC(=O)Cc2cnsc2)=O)c(C)o1 CCCC(O)CC(=O)NCC1CN(C(=O)Cc2cnccn2)CC1O c1(C(=O)Nc2ncc(CSc3ccc(F)cc3)s2)ccc2c(c1)COCO2 N#CC1(C(N2CC(NC(C3CCCSC3)=O)C(O)C2)=O)CC2C=CC1C2 C1(C(N(CCCCCNC(C2CCN(C)C2C2CC2)=O)C)=O)CN2CCN1CC2 N1(C(COc2cccc(CC)c2)=O)CCCC(NC(=O)CS(N)(=O)=O)C1C C(C)(C(=O)N1CC2CC1C2NC(c1ccsn1)=O)(C(C)C)OC C(C)(C)(CC(=O)O)n1cc(C2(N(C(c3csc(C(C)C)n3)=O)C)CC2)nn1 C(=O)(C1CCCc2ccccc21)NCC(CCNC(C1(C)CC=CCC1)=O)OC N1(C(CC(C)(C)NC(C2CC3(CC3)C2)=O)=O)CC2OCCOC2C1 N1(C(CC2ON=C(CC)C2)=O)CC2=C(C1)CN(C(c1ccc(C(F)F)cc1)=O)C2 c1(N2CCCC(C(N)=O)C2)nc(=NCC2(c3ccccn3)CC2)[nH]c2ccsc12 Cc1cc(NC(c2ccc(C(C)(C)F)cc2)=O)cc(C#N)c1 c1(C(N(C(C)C(=O)NCCC(C)C)CC)=O)ccc2ccoc2c1 CC1(C)C(=O)CC1C(=O)NC1(CCC(=O)Nc2ccc(C3CC3)cc2)CCCC1 N1(C(CCOCCNC(=O)C(CO)C(F)(F)F)=O)CCCC12CCNC2=O N1(C(c2n(C)ncc2)CNC(C2CC(C)(C)CO2)=O)CC2(CC(N3CCCC3)C2)C1 C1(C(=O)NCC2(F)CN(C(C(C)(C)OCC)=O)C2)CCOC(C(C)C)C1 C1(C)(CC(N2CC(CNC(C(C)SC(C)C)=O)C2)=O)CC1(Cl)Cl N1(C(C2C(C(=O)OC)CC2)=O)CC2CC1CC2NC(=O)CN(C)C(C)C CC(C)CC(O)C(=O)N1CCC(CC(=O)NCCCN2CCCCC2)C1 c1(OC)ccncc1C(=O)NC(C1(O)CCN(C(c2ccc(F)s2)=O)C1)C C(CO)(CCCCNC(=O)CS(=O)(=O)NC)NC(c1ncc(CC)nc1)=O c1(C(=O)NC2CC(O)(CNC(CC(=O)NCC#C)=O)C2)ncccc1O CC(C)=C=CC(=O)NC1(c2cc[nH]c2C(=O)NC2(C)CCCC2O)CC1 c1(C(=O)NCC2C(C)(C)CCCC2)n[nH]c2c1CN(C(=O)CC1CCCOC1)C2 c1(C(C)=O)cc(C(=O)NCC2C(C)CCN2C(=O)Cn2cnnn2)cnc1C c1(-n2cc(NCC3(C(=O)O)CC(OC)C3)nn2)c(Cl)cccc1Br n1(CC(N2C(CC)CN(c3ccccc3)CC2)=O)ccc(=O)c(O)c1C c1(C(=O)NC(C)CC(C)NC(c2cccc(F)n2)=O)cc(Cl)ncc1Cl C1(C)(CNC(c2cnn(C)c2C(F)F)=O)CCc2ccccc2C1 N1(C(c2c(CC)scc2)=O)CCC2(CC2NC(=O)CC(C)c2ccco2)C1 C12CCN(CC(C)(C)C1)C=CCN2.C1(C)(c2c(C)nsc2N)CCN(C)C1=O c1(-c2nnc(N(CCSCC(C)C)CC)n2CC(C)C)c(F)c(F)c(F)c(F)c1F n1(CC(=O)NC(C)CNC(C2CC(C)(F)C2)=O)nc(C(F)F)cc1C1CC1 Cc1n[nH]c2cnc(C(=O)NCC3CCN3C(C3OCCOC34CCC4)=O)cc12 C1(CNC(CCC=C(C)C)=O)CCC(C)CN1C(=O)CCc1ccn(C)n1 C#Cc1cc(C(=O)NC2COCC2NC(=O)CC2CC2(C)C)ccc1C c1nc(C)c2c(n1)CCCC2.C1(N(CCNC=O)CC)COC2(CCCNC2)C1 CC1CN(C(C2CC2F)=O)CCCN1C(=O)C(Cc1ccc(Cl)cc1)CO Cn1nnc2cc(C(=O)NCC3CCN3C(C3CC=CCO3)=O)ccc12 C12(C(=O)NC3C4CN(C(COC(C)=O)=O)CC43)CC3CC(CC(C3)C1)C2 N1(C(Cc2c(CC)cccc2CC)=O)CCOCC2(CCC2)C1 CC1CCC(CC(=O)NCC2(O)CN(C(C3CC34CC(O)C4)=O)C2)OC1 C(C(=O)NOCc1ccc(C)cc1)(C1CCOCC1)NC(c1nc(CC)oc1)=O C1(CNC(CCOCCC)=O)(CNC(c2ccc[nH]2)=O)CC12CCC2 C1(C(=O)NC(C(=O)NC)C2CC2)N(C(=O)C=C(C)C(C)(C)C)CCC1(C)C c1(C(N2CCC(C)(CCNC(C3N(C)CC(O)C3)=O)C2)=O)nnn2c1CCCC2 c1(CCC(N2CCC(O)(CNC(CN(C)C)=O)C2)=O)cc(F)ccc1Br c1(CCCC)ocnc1C(=O)N(CCCNC(=O)CCC1CCC1)C1CC1 n1(CC(N2CCC(OCCNC(C(CC)(C)O)=O)C2)=O)nc(C)c(Cl)c1C c1(CCCNC(c2cnc(CC)s2)c2nnnn2CC)ccc(C)cc1 CC1CCN(c2cc(C(F)(F)F)nc(Cl)n2)CC1NC(c1ccc(F)c(Cl)n1)=O C1(C(N(C2CC(=O)N2)CC)=O)CC2CC1CN(C(=O)C=CC1CC1)C2 c1(OC)cc(C)c(C(C)NC2(c3nnnn3C)CCC3(CC2)CC3)cc1OC(C)=O Cc1ccc2c(c1)Nc1scc-2n1.c1(COCc2cnn(C)c2)ccccc1 CC(C)(C)CCCC(=O)N1CCC(CO)(NC(=O)CCC2CNC(=O)N2)C1 CC1CCC(NC(=O)CCNC(c2ccco2)=O)CN1Cc1ccnc(Cl)c1 Cn1ncc(C2CC2)c1C(N1CC(=C(F)CNC(=O)Cc2csc(S)n2)C1)=O N1(C(C(CSC)C)=O)CCN(C(=O)C(O)CCC2CC2)CC1C1CCC1 O=C(C1=C(Cl)CCOC1)N1CCCN(C(C2C3CCCCC23)=O)CC1 CC1=C(C(=O)N(C2CC(NC(=O)C(C)OCC3CC3)C2)C)SCCO1 C1(C(=O)NC2CCCN(C(c3c(OC)csc3)=O)C2)CCc2ncsc2C1 Cc1nsc(NC2CC2CNC(=O)CCc2csc(=N)[nH]2)c1C(=O)NC1CC1 Cc1cc(F)c(C(N2C3CCC2C(CNC(c2coc(CO)c2)=O)C3)=O)c(F)c1 C1(NC(C2CN(C(N)=O)C2)=O)CN(C(c2csc(O)n2)=O)C2(CCOC2)C1 CS(=O)(=O)c1ccnc(NC2CC(NC(c3cnn[nH]3)=O)C2)n1 c1(C(N(CCNC(c2c(COC)cco2)=O)CC2CC2)=O)ccc(Cl)cc1C c1(C(=O)NCC(CN(C(COCCOCC#C)=O)C)C)cc(C2CCCC2)no1 N1(C(c2cnc(CC)s2)=O)CC(O)C(O)C1CNC(c1ccc(CO)c(F)c1)=O n1(CCCOC)nnnc1C(CCSC1CCCC1)NCc1cc(C2CC2)cs1 c1(C(=O)NC2CC3CN(C(C(CC)(C)C#N)=O)CC3C2)c(F)c(F)cc(F)c1F c1(C(=O)NCC2C(NC(c3c(CCC)nns3)=O)C2)csc2c1CCC(C)C2 CC1(C)CCN(C(c2ccccc2)C(=O)NCc2ccc(F)cc2)CCS1(=O)=O Cn1ncc(C(N2CCN(C(=O)NCc3ccco3)CC2)=O)c1Cl CC(C)(CCCNC(=O)CN1CCOC1=O)NC(C1CCCC(F)C1)=O C#Cc1ccc(NC(C2CCOC2CNC(C2(F)C(C)(C)C2(C)C)=O)=O)c(C)c1 c1(C(N(C2CCCN(C(c3cn4ccsc4n3)=O)C2)C)=O)cnn(C)c1C#N C(=O)(C(CN(C)C)CC)NCC1(F)CC(CC)C1.c12cc(on1)C(=O)N2 C(=O)(C1CCCc2ncccc21)NC(CNC(C1(CCCC)CCC1)=O)C(C)C C(=O)(CCCC(=O)NCCC1CCC(NC(c2cc(O)ncc2F)=O)C1)N(C)C c1(C(=O)NCC2CC(NC(C3ON=C(C)C3C)=O)C2)ccc2[nH]c(=N)n(C)c2c1 C(=O)(C(CC(C)C)C(N)=O)NC1C2CC(CNC(Cn3ccc(C)n3)=O)(C2)OC1 C1(CNC(C(C(C)(C)C)C2CCC2)=O)CN(C(C2CCC(=O)N2)=O)CCC1(F)F N1(C(c2c(CC)noc2)=O)CC(C(=O)NCc2nc(=O)o[nH]2)C(C(C)C)C1 c1(CNCCCCc2ccc(OCC(=O)N(C)C)cc2)c(F)ccc(O)c1O C(N=c1[nH]c2c(c(=NC3CC4CC34)[nH]1)CCCCC2)C1CCCN(CC)C1 c1(COC(C(CC)c2ccccc2)=O)cccc([N+](=O)[O-])c1 C12(NC(N(CC(c3ccccc3)(C)O)C)=O)CCCC1C2(F)F n1(CC(=O)NC2CC(O)(CNC(=O)CC#N)C2)nc(C(F)(F)F)cc1C1CC1 C1(C(=O)NCC2C(NC(CCSC)=O)COC2)Cc2ccccc2O1 C1(C(=O)NCC2CCOCC2)COC2(C1)CN(C(=O)CC1CC3CCC1C3)C2 C(=O)CC1CCOc2ccccc21.CC1(C)CCOC1c1ccc(-c2nn[nH]n2)cc1 C(=O)(C(F)CC(C)(C)NC(=O)CCc1cncs1)NCC(C)OCCO c1(CCN(C(=O)CCc2ccncc2)C(C2COC2)C2CC2)ccccc1Cl C1(NC(CN(C(CNC(C)=O)=O)C2CCC2)=O)CC2CC1OC(=O)N2 c1(C(=O)NC(C(=O)NCC(CC(C)C)N(C)C)c2ccco2)cccc2[nH]ccc12 n1(CC)cc(C(N2CCC(OCCNC(=O)CNS(N)(=O)=O)C2)=O)c(C2CC2)n1 C12(C(N(CC#C)CCF)=O)CC(C)(CN1C(c1cccc(COC)c1)=O)C2 CC(C)C#CC(=O)N1CC(C(C(c2ccccc2)=O)NC(=O)CCC2CC2(F)F)C1 C1(C(=O)NC2(C)CN(C(c3c(C)nc(O)[nH]3)=O)C2)Cc2cccnc2C1 C1(C)(CC(=O)NC(CC)(C)CNC(=O)C=C2CCC(C)C2)CCCCC1 C1(CNC(c2cc(OC)n[nH]2)=O)CN(C(C2CC2F)=O)CC1O N1(C(c2cnc(S)nc2)=O)CCC(O)(CNC(=O)CCNC(C2CC2CF)=O)C1 c1(C(N(CC(CC)NC(C2CCCN2C(C)=O)=O)CC)=O)nnn(C)n1 CCC(C)C(C)NC(C1(CCNC(=O)C(C)(C2(C)CC2)OC)CC1)=O C(=O)(C(CC(C)C)CC(C)C)N1CCN(C(c2nn(CC)c(O)c2)=O)C2C1C2 c1(C(N(C(C(CC(=O)OC)C)=O)C2CC(S(C)=O)C2)=O)ccc(S(C)(=O)=O)[nH]1 Cc1cc(C(=O)N(CC(C)CNC(=O)C(C)Oc2cccc(F)c2)C)cnn1 Cc1ncc(C(N2CC3(C2)CN(C(c2cccc(C(F)F)n2)=O)C3)=O)c(=N)[nH]1 C1(CC(=O)N(Cc2cnn(C(F)F)c2)CC2CCCC2)CCC2CC12 C1(C(C)NC(=O)CNC=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1 C1(NC(COCC=C)=O)CC2CCC(C1)N2C(c1ncn(C)n1)=O c1(SC)ccc(C)c(C(N2CCCC(C)(NC(=O)C=CCN(C)C)C2)=O)c1 c1(C(=O)NCC(COC)NC(C2CC3(CC3)CO2)=O)onc(C)c1CO c1(NC(c2ccc(Nc3c(F)cnc(C)n3)nc2)=O)cc(F)c(O)cc1Cl C(=O)(C(O)(C(F)(F)F)c1cn(CCC2CC2)nn1)N(C(C1CCC(=O)NC1)=O)CCO C1(CC(N2CCN(C(CCCOC(C)=O)=O)CC2C)=O)Cn2ccnc2NC1=O CC(C(C)(C)NC(=O)C(F)=C1CCC1)NC(c1cc(C2CC2)ns1)=O Cc1cc(F)c(CNC(=O)N(C)CCC2CCCN(C(=O)C(C)(C)C)C2)c(F)c1 c1(-c2nc(C(C)SCC)nn2-c2ccccc2Cl)coc(S(N)(=O)=O)c1 Cc1cnccc1C=CC(=O)NC1CC(C)(CNC(=O)C(C)CO)C1 c1(C(C)C)cccc(F)c1C(=O)NCC12CC1CN(C(c1c[nH]c(=N)o1)=O)C2 CN1CC2C(C(=O)NC3(CNC(=O)CC4(C(F)(F)F)CNC(=O)C4)CCC3)C2C1 CC(F)CC(=O)NC(C)(CNC(=O)CCC1CCC1)C1CCC1 N1(C(c2cc(C)nn2CCO)=O)CC2CCC1CN2C(=O)Cc1ccc(F)cc1 c1(CNC(c2c(C)onc2-c2ccc(Cl)cc2F)=O)ccnc2c1CNCC2 C1(C(=O)OC)CC12CCN(C(=O)N(C(C(C)C)C(C)C)C1CC1)CC2 C(=O)(N=c1[nH][nH]c2c1CN(C(=O)C(Cl)(Cl)Cl)C2(C)C)c1cccc(C)n1 C(=O)(C(C)(C)CC(=O)N1C2CCC(C2)C1CNC(=O)Cc1ccoc1)OCC c1(C(N2CCC2Cn2cc(-c3ccc(CO)cc3)nn2)=O)cccn2ncnc12 C(=O)(CCCN=[N+]=[N-])NC(CCCCNC(Cc1cccc(C)c1)=O)C Cc1cc(C(=O)NC2CCC2NC(c2ncoc2C2CC2)=O)c2nc(C)n(C)c2n1 C(=O)(C1Cc2ccccc21)NCc1cccc(CNC(c2c(CC)onc2)=O)c1 C12CC3(CC3)CN1C2=O.C1(C)(CNC(Cc2nc(C)[nH]n2)=O)CNC(=O)O1 C1(c2nnnn2-c2ccccc2C)(NCC2CC(OC)C2)COCC(C)(C)C1 C1(C(=O)NCC(COC)NC(=O)C(C)(C)C2CCOC2)CCCCS1(=O)=O N1(C(C(C)SCC)=O)CC2CN(C(c3cccc(C)c3F)=O)CC2(C)C1 N1(C(CN(CCC)C(C2CCCCO2)=O)=O)CC(CN(C)C)CC1(C)C C1(CNC(CC2C(C)(C)CO2)=O)CCCC(NC(=O)CC(=O)Nc2ccc(=O)oc2)C1 C1(NC(C2CC(=C)C2)=O)CCOC2(CCN(C(=O)CCC(C)CN(C)C)CC2)C1 C1(CNC(=O)Nc2nc(Br)cc(OC)n2)CCC(C)(C)C(=O)N1 C(C(C(F)(F)F)N1CCNCC1)N(CC(=O)Nc1nn[nH]n1)C C(=O)(C1=C(Cl)CC1)NCC1(C)CC(NC(c2n(CC)ccc2)=O)C1 CC1CC(C)N(C(c2cccn2C)=O)CCN1C(=O)Cc1ccsc1 N1(C(CC(C)OC)=O)CCC2CN(C(=O)CCc3cncs3)CC2CC1 c1(OC)cnc(C(=O)NC2(CO)CCN(C(c3cc(C(C)C)on3)=O)C2)nc1 C1(C(=O)NCCC(=O)NCCCNC(=O)CCN2CCOC2=O)CC2CC1C2 N1(C2C(CNC(c3cnn(C(F)F)c3)=O)C2)CCc2ccccc21 N1(C(C2OCCN(C(C)C)C2)=O)CC2(CCCC(CNC(=O)C3=CCCC3)O2)C1 N#Cc1cc(C(N2CCCC2C2(O)CN(C(C3CCCS3)=O)C2)=O)co1 C1(N(C(c2ncn(CC)c2)=O)C)C2CN(C(=O)CCc3ccncc3)CC12 CON=CC(=O)NCC(c1ccccc1)CNC(C1CC(=C2CC2)C1)=O c1(CC)nc(CNC(C2CCOC2CNC(=O)C(C)(C)n2cncn2)=O)cs1 n1(CCC(=O)NC(C2CN(C(C3COC3)=O)CCO2)C)ncn(C)c1=O C1(CNC(C2(C)CC2)=O)CCC2(CO1)CC(NC(=O)CCc1cc[nH]n1)C2 N1(C(CC2(C#N)CCOCC2)=O)C2CCCC1CN(C(=O)CCCCC1CC1)C2 CC(C)CCC(O)C(=O)N1CCC(N(C(=O)C=Cc2ccncc2)C)CC1 Cc1cc(C)c(CCNC(=O)C(CC(C)C)ONC(c2ncc(F)cn2)=O)c(C)c1 C1(NC(CN(C(C)C)C)=O)CC2CC(C1)N(C(C1CCCC(=O)C1)=O)C2 C1(C(=O)OC)CCCN(C(c2nccnc2OC(F)(F)F)=O)C1 N(C1CCCc2cc(F)ccc21)C(C1C(CN(C)C)CCCC1)=O Cc1cncc2c(C(=O)NCC3CC(O)CN3C(=O)CC3CCOCC3)cnn12 N1(C(c2c(C)cc(C)s2)=O)CC2CC(NC(=O)C#CC3CCCO3)CC1C2 C1(CCC(=O)NCC(C2CCCCO2)(C)C)CCC(NC(=O)Cc2cn[nH]c2)C1 Cc1cc(CN2CCC(c3nncs3)C2)c(F)c(Br)c1 c1(OC)cc(C(N2CCCC2CNC(c2cncc(C)c2)=O)=O)cc(F)c1 Cc1cc(C)c(C(=O)NCC2CCCN2C(=O)CCc2ccccc2Cl)c(C)n1 N1(C(=O)C=Cc2cccs2)CCC2(CCN(C(c3ccn(C4CC4)n3)=O)CC2)C1 CC1CN=C2NC(C(=O)N3CC(N(C)C(c4cc(C(C)(C)C)no4)=O)C3)=NN2C1 C#Cc1cc(C(=O)NCC2(O)CC(C(N3CCOC(C)(CC)C3)=O)C2)ccc1C N1(C(CN(C2CCC(NC(=O)Cc3ccns3)C2)C)=O)CC(F)CC1CO NS(=O)(=O)N1CCCN(C(=O)C(N2CCN(Cc3cccc(Cl)c3)CC2)=O)CC1 CC(C)CC(CNC(=O)CCCCCNC(C1(N(C)C)CC1)=O)CO c1(C(N(C)CC2CN(C(=O)CC3CC(CF)C3)CCO2)=O)cc2cccnn2c1 N1(C(CS(CCC)(=O)=O)=O)CC23CCCC2(C1)CN(C(C1CCOC1)=O)C3 Cc1cc(N2CCN(C(c3ncccc3F)=O)CCC2C)ccc1[N+](=O)[O-] N1(C(c2[nH]cc(C#N)c2)=O)CCC(NC(c2cc(Br)ccn2)=O)C(O)C1 C1(NC(CSCC#C)=O)CN(C(c2cc3n(n2)CC(F)C3)=O)C2(CCCOC2)C1 c1(N2CCC(CC(N3CCN4CCC3CC4)=O)C2)cc2ncnn2cn1 N1(C(C(C)Oc2ccccc2)=O)CCCCC(NC(c2ccc(C(N)=O)o2)=O)C1 N1(C(=O)CCc2ccc[nH]2)CCC2CCN(C(C34CC5CC3C4C5)=O)CC12 Cc1nc(O)c(C(=O)NC2CCCCN(C(=O)Cc3ccoc3)C2)nc1C c1(C(N2C3(CC(COC)C3)CC2)=O)nc2c(Br)cncc2[nH]1 N1(C(C(=C)C)=O)CCCOC(CNC(C23CC2CCCN3C(=O)OC(C)(C)C)=O)C1 N1(CC(=O)N(CC(C)NC(c2cc(C(=O)N(C)C)co2)=O)C)CCCCC1=O Cc1noc(C)c1Nc1nccc(N2CCCCCC2)n1.C12CCCC1NCC2 Cc1cc(C(N2CC(CNC(=O)Cn3ccnn3)CCC2C)=O)cc(C)c1 C(C)(C)(C(C)CC(=O)NCC(C)CC1CC1)NC(c1cc(COC)oc1C)=O c1(C(=O)NC2CCCCC2NC(C2CCCC23CCC3)=O)cc2n(n1)CCCC2 C(CCCC(=O)N(C)CCOCCCN(C(=O)CN(C1CCSC1)C)C)SC N1(C(C(C(C)(C)C)CO)=O)CCC2CCC(C1)N2C(=O)CCOC1CC(F)(F)C1 c1(OC)c(CCn2c(C3CC3)nnc2S)cc(C)cc1C C(C(=O)NCC1CCCCN(C)C1)(C(C)(C)C)NC(c1cc(C(C)C)n(C)n1)=O C1(NC(Cn2c(C)cc(C)n2)=O)CN(C(c2cccs2)=O)C2(CCC2)C1 N1(C(C(C)S)=O)CCC2(CCCC2C(N2CCNC(=O)C2)=O)C1 N1(C(CCc2onc(C)n2)=O)CCC2CC12C(N1CC(CCCCN(C)C)C1)=O c1(C(=O)NCCN(C(c2ncc(C)c(C)c2)=O)C)c(C)nc2sc(C)nn12 C1(CNC(c2n(C(C)C)ccc2)=O)CC(N=c2[nH]c3cc(Br)ccc3o2)C1 c1(OC)cc(Cl)ccc1C(N1CCC(C)C1CNC(=O)C1=CCCS1)=O N1(C(CNC(N)=O)=O)CCC2(CC1)CCN(c1ncc(F)c(-c3ccsc3)n1)CC2 NC1CC2CCCC(C1)N2S(=O)(=O)c1cnccc1N1CCC(CCO)C1 c1(OC)ccccc1C1(NC(=O)NCCNC(C2SC3C=CC2C3)=O)CC1.CC C1(CC#C)CN(C(N2CCC(OCc3ccccc3F)CC2)=O)CCO1 C(CN=c1[nH]c2ccccc2s1)N1CC(C)OC(C)C1 CCCCCC(F)C(=O)N(C)CC1(C(=O)Nc2ccn(CCCC)n2)CC1 CCC(C)(C(=O)NCc1c[nH]nc1C(=O)NC1CCC(C(=O)NC)C1)OC c1(CSC)cc(CCNC(=O)CC2(C)CCN2C(=O)C(CC)N(C)C)on1 CCC(CC(F)(F)F)C(=O)N1CCCC(Nc2ncnc(C)c2C#N)CC1 c1(C(C(=O)OC(C)(C)C)(C)C)ccc(F)cc1F.C1(OC)C(=O)N2CCC12 N1(C(c2cccc(C)c2O)=O)C2CCC(C(=O)N(C)OC3CCCC3)C1CC2 c1(OC)ccc(C(=O)NC2CC(C(=O)NCCc3ccncc3)C2(C)C)nc1 C1(O)(CNC(c2cnc(C3CCCO3)s2)=O)CCCN(C(=O)C2CC2)C1 C(=O)(CC(C)CCC)NCCCN(C(C1C2CCC1(c1ccco1)C2)=O)CC C=CC1(C(N2CCCC(CCCO)C2)=O)CCN(C(=O)Cc2cc[nH]c2)CC1 C1(CNC(CN(CC)CC)=O)C(C(N2CC=CC2CF)=O)C1(C)C C1(C(=O)NC2(CC=C)CN(C(=O)C(C)CCOC)C2)CCOC(C)(C)C1 N1(C(=O)COC2CC=CC2)CC23CCCC2(C1)CN(C(=O)CC1CCCCO1)C3 c1(C(N2CC(NC(CCOCC#C)=O)C(C)C2)=O)cc(C2CC2)nc(O)c1 Cc1cc(C(N2CCCC(C)(CNC(c3cc(C)n(C)c3)=O)C2)=O)ccc1O CCC(CC(=O)NCC1CC(OC)CN1C(c1cn(C(F)F)c(C)n1)=O)C(F)F C1(CNC(CC2(COC)CC2)=O)CC2(CCN(C(=O)C(C)(C)SC)CC2)CO1 N1(C(=O)Cc2cccc(O)c2)CCCCC(F)(F)C1.CC12C=CCN1C2=O C1(C(=O)NC(COC)C2(C)CC2)CN(C(=O)Cc2cnccn2)CCO1 C1(NC(C(C2CC2)NC(CC#N)=O)=O)CCOCC1 CC1(C)C(NC(c2ccc(C3CC3)nc2)=O)CC1CNC(=O)CCc1cccnc1 c1(C(=O)NCC(C)N(C(COCc2cc(C)no2)=O)C)cc(C)sc1C C(=O)(C1=CCc2ccccc21)N1CC2(OCC(NC(C(CC)=CC)=O)C2)C1 CN1CCCC(F)(C(=O)NCCCC2CCCN2C(=O)CCCn2cncn2)C1 CCC(C)(C)C(O)C(=O)NCC1(C)CCCN1C(c1cncn1C)=O CC(C)(CC(=O)NC1CC(COc2cc(Cl)cc(Cl)c2)C1)CC(F)F N1(C(C2CCCN(NC(C3C4CC5C(C4)C35)=O)C2)=O)CCSC2(CCC2)C1 c1(C(N(C)CC2CCCCN2C(=O)COC2(C)CCC2)=O)cc2ccccc2[nH]1 C1(C)(C(=O)NC2CC(CCNC(c3n(CCC)ccc3)=O)C2)CCCCNC1=O C1(O)(CNC(C(CSC)OC)=O)CCCN(C(c2sccc2F)=O)C1 C(C(C(=O)N1CCC(NC(c2cnccc2Cl)=O)C1)C(C)(C)C)OCC=C C12CN(CC1c1ccccc1)C(=O)CC2C.C(=O)(CC1COC1)OC C(=O)(CC(C)(O)C(F)(F)F)N(CCCNC(c1ccc(N=[N+]=[N-])cc1)=O)CC Cc1nn(C)c(=O)c(C(=O)NC2COC3(C2)CN(C(=O)C(O)CC2CC2)C3)c1C c1(C(C)=O)ccc(C(=O)NCC(C2CC2)NC(=O)CSC2CC2)nc1 CC1C(NC(c2n[nH]c3ccc(F)cc23)=O)CC2CCC1N2c1nccnc1F c1(C(n2cc(CNC(CCNC)=O)nn2)C)ccccc1[N+](=O)[O-] CC(C)CC(C)CC(C)C(=O)NCC1CCC(CNC(C2CCCSC2)=O)CC1 N1(C(CC2C(C)(C)C2)=O)CCCN(C(=O)COC2CCC2)CC1CO N1(C(C(CC)n2cccn2)=O)CC2CC(NC(=O)C(C)NC(N)=O)CC1C2 C(=O)(CC(CN(C)C)CC)NCC(CCCC)NC(c1c(C)ncn1O)=O c1(OC)ccnc(NC(=O)NC2CCCC(C(=O)NCc3ccccc3)C2)c1F c1(C(=O)NC2CC(CNC(c3cc(C)no3)=O)C2)cccc2cncn12 C(=O)(CS(=O)(=O)c1ccc([N+](=O)[O-])cc1)NCCCNC(=O)Cc1cccs1 Cc1nsc(C(=O)NC(CCN(C)C)C(=O)NCc2ccnn2C)c1N C(=O)(C(F)(F)C(O)C(C)C)NCCN(C(=O)Cc1cccc(OCC(F)F)n1)CC c1(C2C(CC(N3CCC(c4ccc(F)cc4)C3)=O)C2)ccccc1F C1(NC(C(CC)OC)=O)CN(C(=O)CNC(C)=O)CC2(CC2)C1 Cc1c(C(=O)NCC2CC2CNC(=O)CC(=O)N(C)C)oc2ccccc12 c1(C(=O)NCC(=O)OCC)ncccc1CC.c1(N)ccsc1 c1(C(N2C(CNC(C3(F)CCOC3)=O)CC(OC)C2)=O)cc2cccnc2s1 c1(CCN=C(NC(c2csnn2)C)NCC2CCOCC2)nc2c(s1)CCCC2 CC(C(C)(C)C(=O)NC1(C2CC2)CCOC1)NC(=O)COCC1CCCC1 c1(C(N2CCOC(CC)C2)C(=O)NCC=C)cc(Cl)c(F)c(Cl)c1 Cc1cc(F)cnc1C(=O)NCC(O)C(=O)N(CC(C)(O)C1CC1)C c1(NC(C2N(C(c3cn(C4CC4)nn3)=O)CCC(=C)C2)=O)ccc(C)c(C#N)c1 C1(NC(C(CCC)C#N)=O)CC12CCN(C(c1oc(CO)nc1C)=O)CC2 CC1(NC(C2CC23CC(NC(=O)CCCN=[N+]=[N-])C3)=O)CN2CCC1CC2 c1(C(=O)NC(C2C(C(N(CC(O)CO)CC)=O)C2)C)ccnn1C Cc1c(C(=O)NCC2(CO)CCN(C(=O)CN3CC=CC3)C2)ccn1C1CC1 c1(NC(C(COCC)N(CC(F)Cl)CCC)=O)ccccc1Br c1(CNC2(COC)CSC2)cc(OCC(F)F)ccc1C CC1CCC(NC(c2cccc(F)c2Cl)=O)CN1C(C12CC(C1)C2)=O c1(NC(N(C)Cc2nc(C(C)OC)sc2)=O)cc(F)ccc1C(C)C N1(C(c2n(C)nc(O)c2)=O)CCCC(C(=O)NC2(C)CCCC2)CC1 CC1CC(NC(C2CC3CC3C2)=O)CN(C(c2nc(C(F)(F)F)ccc2N)=O)C1 CN1CC(NC(=O)C(=O)NCC(c2c(Cl)cccc2Cl)O)CC12CCCC2 C1(O)(c2c(OC)ccc(C)c2)CN(N2CCCC2CCC(C)C)C1 N1(C(Cc2cc(C)on2)=O)CCCCC(C(=O)NC2COC(=O)C2)C1 c1(C(=O)NCC(O)CNC(c2cn3ccsc3n2)=O)ccc(CO)c(Cl)c1 c1(CC)ccc(F)c(C(N2CC3CCCC2C3)C(=O)NC(C)CC)c1 C(=O)(NNC(=O)c1ccc(OCC(N)=O)cc1)c1nc(CC)[nH]n1 CCC(CCCC(=O)NC1(CO)CCC1)NC(c1cnn(C2CC2)c1)=O N#Cc1cnc2ccc(Br)cc2c1NC(C1CCc2ncc(Br)n2C1)=O c1(-c2cc(C)on2)cc(Cl)cc2c1NCCC2 N1(C(C2N(C(Cc3nc(C)oc3)=O)C(C)C2)=O)C2CCCC1CC2 c1(-c2cn(C3(O)CCN(C(C(CC)C)=O)CC3)nn2)oc2ccccc2c1C c1(C(=O)NCCOCCNC(C(C)(C)c2cccnc2)=O)ccc(Cl)cc1 C1(NC(CCCCOCC(C)C)=O)CC(C)CN(C(C23CCCC(CO2)C3)=O)C1 c1(NC(N2CCN(CC(=O)NCCCO)C(=O)C2)=O)c(F)c(F)c(F)c(F)c1F c1(C(=O)NC2C(NC(C(CCC)C(C)C)=O)C2)cc2c(nc1O)CC(C)(C)CC2 CC1=C(C(=O)NCc2ccoc2C(N(C)CP(C)(C)=O)=O)COCC1 c1(C(=O)NC2C(NC(=O)Cc3ccc(O)cn3)CC2)nnc2n1CCCCC2 Cc1c(O)c(=O)ccn1CC(N1CCC2(NC(=O)CCc3cc[nH]n3)CC2C1)=O C1(c2nnnn2C)(NCCc2c(C)cccc2)CC2OC(C)(C)OC2C1 C1(C(=O)NCC(COC)O)CCCCCCN1C(=O)CC1CCCCC1C N1(C(C2N(C(CCOC)(C)C)CCC2)=O)CCC(Oc2cccnc2)CC1 CN(C)S(=O)(=O)N1CCCC(CNC(C2(C)CC(N)CCO2)=O)C1 c1(CC)ccc(C(=O)NC2CCCC2C(=O)NCCC2CCCC2)nc1 N1(C(C2C(NC(C3(CN(C)C)CC3)=O)COC2)=O)CCN(C)C(CO)C1 C(C(C(C)C(C)C)NC(=O)C(C)(C)C1CC1)NC(COCc1ccc(C)s1)=O c1(CC)ccc(N2CCCC2)c(C(=O)CN(CC)CC2CCCS2)c1 N1(C(C(C2CCC2)OC)=O)CCC(F)(CNC(=O)C(=C2CCCCC2)F)CC1 C(=O)(CC1=CSC2=NCCN12)NCC(C)NC(=O)CC1CCCOC1 N1(C(C2(C#C)CCC2)=O)CCCC(NC(=O)C(c2ccccc2)SC)C1 C1(CC(=O)NC2C=CCN(C(C3CCSCC3)=O)C2)CCCC12CC2 c1(NC(=O)OCC)cc(NCC(F)(F)F)ccc1C.c12ccnc(c1)C(=O)N2 CCCCCCCCCn1cc(C2CC(O)CN2C(=O)C(C)(O)C(C)C)nn1 C12(C(=O)NCC3CC(C)(C)N(C(C4(O)CCOCC4)=O)C3)CCCN(CCC1)C2 C(=O)(C(F)C(F)(F)F)NCC1CN(C(C(=O)NCCNC(C)=O)=O)C(C)C1 N1(C(=O)CC2(C(=O)OC(C)(C)C)CC=CC2)CCC(=O)C2(CCC2)C1 CC1CCN(C(C23CC(CN2C(C2C4CN(C)CC24)=O)C3)=O)C1CO Cc1c(Br)ccc2nc(NCc3cscn3)nn12.c12ccnc(c1)CNC2=O c1(C(N(C)CC2(O)CN(C(=O)CCN3CCC(F)C3)C2)=O)cnc(S(C)(=O)=O)s1 S(=O)(=O)(c1ccc2[nH]c(=NCC3CCCCO3)sc2c1)NCC1(CC)CC1(C)C c1(SC)cccc(CC(=O)N(CC2(F)CC2)CC2CC2)c1 C#Cc1cc(C(=O)NC2CC3CCC2N(C(=O)CC(O)CC)C3)cc(F)c1 N1(C(c2cc(C)c(N)cn2)=O)CC2CC3CC2C1C3NC(=O)Cc1cc[nH]n1 C(=O)(C(F)C(C)(F)F)N1CCC(CC=C)(C(=O)NCC2CCCC(O)C2)C1 CCCC(C(=O)N1CC(C2CC2)(C(=O)N(C2CC(OCC)C2)C)C1)C(C)C Cc1cc(C(=O)NC2(CF)CCN(C(C3CC(C)CCO3)=O)C2)cc(C)c1 c1(OC)cc(N)ccc1C(=O)NCCC(C)N(C)C(C12CCCC(CO1)C2)=O CN=c1[nH]cc(C(=O)NC2CCN(C(=O)C(C)(C3CC3)OC)CC2)s1 C1(C(=O)NCCCCCC#C)C2CCCC2CN1C(=O)C(O)CN(C)C c1(C(N2C(CNC(C3(C#C)CCC3)=O)CC2)=O)cc(Cl)ccc1O C1(NC(CC)=O)CCN(C(=O)C=Cc2cccs2)CC1C C1(CNC(C(C=C)C)=O)CCCCN(C(=O)C(C)=CC(C)(C)C)C1 C1(NC(=O)Cc2cnc[nH]2)CC2CCC1C(NC(C1(CCF)CCOCC1)=O)C2 Cc1nn(C)c(Cl)c1C(=O)NCC#CCNC(C1(Cl)CC1)=O c1(OCC(=O)NCC2C=CC(NC(=O)CC3(C#N)CC3)C2)ccc(CO)cc1 c1(C(=O)NCC(n2cc(CC(O)C3CC3)nn2)C)cc(N2CCCC2)nc(Cl)c1 c1(CC(=O)NC2(C)CN(C(C(C(CC)O)C)=O)C2)coc2c(F)c(F)ccc12 c1(C(=O)NCC(C2CC2)OC)ccc(-c2ccc(-c3nnc(C)o3)cc2)nn1 C1(OCC)CCc2nc(N(CC(C)OC)C)nc(N3CCC(C)(OC)CC3)c2C1 C1(C(=O)NC2CCCCN(C(C3(C#C)CCC3)=O)C2)CC2(C1)CC(F)(F)C2 N1(C(Cc2cnc(C)s2)=O)CC2(C1)SCCC2NC(c1cc(C(F)F)ncn1)=O Cc1cc(Nc2cc(Br)ccc2NC(C2CC2C(N)=O)=O)nc(C)n1 c1(OCC)ccc(CC(=O)NCC(C)NC(=O)CCNc2ccc(N)cc2)cc1 c1(C(C(=O)NC(C(=O)N(CCCOC)C)C)O)cncn1C C1(NC(CC(C)(C)NC(c2ccc(C#N)s2)=O)=O)CC12CCOCC2 N(C(=NCCCF)NC1CCCn2nc(C)nc21)CC1(CC)CCOCC1 N1(C(C=NOC)=O)CCC2(COC(CNC(c3cc(C)c(C)s3)=O)C2)C1 C1(F)(C(=O)NCC2C(CC(=O)NC(C3C(C(=O)OC)C3)C)C2)CCCCCC1 c1(OC)ccc(Br)c(C(=O)NC(CNC(c2ccn(C)c2C)=O)C2CC2)c1 CC1(C)COC(C(=O)NCC2(C(N)=O)CN(C(=O)CCc3ccc(F)cc3)C2)C1 c1(CNC(C(CC=CCC)C)=O)cccnc1CNC(c1nc(C)oc1OC)=O C1(n2cnnn2)(CC(=O)NC(CCCNC(C(OC)OC)=O)C)CCSCC1 C1(C(=O)OC)CC(C)N(C(c2cc(C(=O)OCCSC)no2)=O)C1 C1(O)(CNC(C2(C)CCCC2)=O)CCCN(C(C2CCN(CCF)CC2)=O)C1 CCC(CC)CC(=O)N(CCC(C)NC(=O)Cn1ccnc1C)C C1(C(F)(F)F)(OC)CC(CNC(=O)C(C)O)(NC(=O)Cc2cnc[nH]2)C1 C(CCF)(C(=O)NCCCc1nc[nH]n1)NC(c1ccc(O)nc1)=O Cc1cnccc1C=CC(=O)NC1(CN(C)C(C2(C)CCCC2O)=O)CC1 C(=O)(C#CC1CCCOC1)N1CCCN(C(Cc2ccc(C)c(O)c2)=O)CC1 N1(C(C(CCSC)N(C)C)=O)CC2(CCC(CNC(c3cnn(C(C)C)c3)=O)O2)C1 C#Cc1cc(F)ccc1CNC1(CNC(C2CC2F)=O)COC1 c1(C(=O)NCC2N(C(C3ON=C(CC)C3)=O)CC2)cnc2cc(C)ccn2c1=O CCC(CC)(CO)C(=O)NCC(C)(C)OCC(N1CC2(C1)CC(C)(O)C2)=O c1(C(N(CC(C)NC(CCSCCCC)=O)CC)=O)cn(C)nn1 C#CC1(O)CC(C(=O)NC(C2CCCCC2)C(C)NC(C2CC3CC3C2)=O)C1 c1(C2(C(=O)NC3CC(O)(CNC(C(F)=CCC)=O)C3)CC2)cc(F)ccc1F C(=O)(C(O)Cn1cncn1)NCCN(C(C(C)N1CCC1)=O)CC1CC1 CCC(CC)(CCNC(c1cc(C2CCCC2)no1)=O)NC(=O)C1CC1 C(=O)(C1=CCc2ccccc21)NCC1(C2CC2)CCN(C(C(F)OC)=O)C1 N1(C(c2onc(C)n2)C)CCC(C2CCCN(C(=O)C(C)C3CC3)C2)C1 N1(C(c2c(C)cccc2C)=O)CCC(C2(NC(C3CNC(=O)CC3C)=O)CC2)C1 c1(OC)cc(Br)cc2c1CN(C(=O)C(=O)NCCC1CCCC(C)C1)CC2 C(C(=O)NCC1CCCN1C(=O)C(C)OCCC(C)C)(C(C)C)OCC c1(C(=O)NCCC(C)N(C(C2C(C(=O)OC)C2)=O)C)ccc(C2CC2)nc1C c1(C(N2CCN(CC(C)NC(C(C=CC)O)=O)CC2)=O)cnc(O)c(F)c1 C1(NC(C2CSC2)=O)(CF)CCN(C(C2(C(F)(F)F)CC2)=O)C1 n1(CC(N2CCCCC2c2cccc(O)c2)=O)sc2cc(Cl)ccc2c1=O c1(C(=O)NCCCC(C)NC(c2coc(CO)c2)=O)ncncc1F C1(CC)CC(N=c2ccc(C(=O)OC)n[nH]2)CCO1.C1(C)(C(F)(F)F)CC(=O)N1 CC1CN(C(c2csc(-c3cnccn3)n2)=O)CC1NC(C1CC(N(C)C)C1)=O c1(C(N2CC(CNC(=O)CCOC3CC3)OCCC2)=O)cnc2ccsc2c1 C(N=c1[nH]c(N2CCN(c3cncnc3)CC2)nc(=N)[nH]1)C1(C)CC2CC2C1 c1(CNC(C(CC=C)(F)F)=O)cnc2cc(Br)ccc2c1 Cc1ccccc1C(N1CCN(CC2(S(C)(=O)=O)CC2)CC1)=O.N12CC(C1)C2=O C1(C(=O)NCC2OCCN(C(C3C(OC)CCCC3)=O)C2)CCCCNC1=O C1(C=C)(C(N(C(C=C)C)C)=O)CCN(C(c2nsnc2O)=O)CC1 c1(C(N2CC3(CN(C(=O)CN4CC5CC5C4)C3)C2)=O)cccc2ccncc12 N1(C(CC2CCC(C)O2)=O)CCC(N(C(=O)COCC2(F)CC2)C)CC1 c1(N)cc(Cl)no1.C12(CCC1)N(C)C2=O.C(=O)(CCOC1COC1)NC1CC1 C(=O)(C1Cc2c(Cl)cccc21)NCC1N(C(c2n(C)ncc2Cl)=O)CC1 CC(C)(CC(F)(F)F)C(=O)NC1CCN(C(c2ccc(Cl)nc2)=O)CCC1CO c1(C(=O)NC(CC)CNC(=O)Cc2cncc(F)c2)cnn2c1CCCC2C c1(C(N2CCC(NC(C(C)=C(CC)C)=O)(CO)CC2)=O)cccc(S(C)=O)c1 CC(C(=O)NC1CCCCN(C(c2cccnn2)=O)C1)C1=CCCC1 N1(C(c2cc(OC)ncn2)=O)CC2CCN(C(C3COC4COCC4O3)=O)C2C1 C1(CCC(=O)NC2CCCC2CNC(=O)COC2CC2(F)F)CCOCC1 C1(NC(c2c(C)ccs2)=O)CCN(C(C2CCC(C)C2)=O)CC1 c1(N2CCC(NC(c3c(C)onc3)=O)C(O)C2)cc2nccn2cn1 N1(C(c2cc(COC)on2)=O)CCC(C(=O)NCC2(F)CCCCC2)(CF)C1 c1(CC)ccc(C(N2CC(NC(C3CC(=C4CC4)C3)=O)CCC2C)=O)cc1Cl C(=O)(C1=Cc2ccccc2OC1)N1CC2CCN(C(CCSC)=O)CC21 N1(C(CCNC(C)=O)=O)CCOC(CNC(c2ccccc2-c2nnc(C)o2)=O)C1 C12(C(N(CCC(=O)NCC3(O)CCSC3)C3CC3)=O)CSCC1C2 C1(NC(C(CC)(C)OC)=O)CCC2CCN(C(c3ccoc3Cl)=O)C1C2 N1(C(C(CC)CC)C(=O)NCCN2CCOCC2)CCCC2(CCN(C)C2)C1 C1(CNC(C2N(CC)CCOC2)=O)CN(C)CCN1C(=O)Cc1ccc(Cl)cc1 C1(CNC(COCCC)=O)CCCC2(CN(C(c3cc(C)ccc3Cl)=O)C2)O1 c1(CN(C(c2ccsc2C)C2CC2)CC)c(F)cc(Br)cc1F N1(C(Cc2n(C)nnc2)=O)CC(C(N2CCOCC(CO)C2)=O)C2(CC2)C1 C=C(C)CC(C(=O)N1CCC(C(=O)Nc2cc(CO)cc(C)c2)C1)OC C1(C(=O)NCC(CNC(CCc2nc(C)sc2)=O)F)CCn2c(C)cnc2C1 S(=O)(=O)(c1ccc(N2C3CCC2c2ccccc23)c(Br)c1)NC1(C)CCOC1 CC(C)CC(F)C(=O)N(CCCOCCNC(C1CC1C(C)C)=O)C C1(O)(CN(CC(=O)Nc2ccccc2Cl)C)CCCN(C(c2sccc2F)=O)C1 c1(C(N(CCC)CCNC(=O)C(C)n2cccn2)=O)cccc(CC)n1 S(=O)(=O)(c1ccc(C#N)c(NCC2CN3CCN2CC3)c1)N(CCN(C)C)C N1(CC(N2CC(C(C)(C)O)(CNC(C=C3CCC(C)C3)=O)C2)=O)CCC(C)(O)C1 C(=O)(C(C)CC(C)(F)F)NCCCC(C)NC(c1c(C)[nH]c(C(C)(C)C)c1)=O CC1CCNCCC1C1(CSC)CC1.c1(NC2(O)CC2)ccc(-c2nccs2)cc1 n1(CC(C)NC(C(C)N(C)C(c2cccc(C)c2)=O)=O)ncc2ccccc12 N1(C(CN2CC(C)C2)=O)CC(CNC(=O)C=Cc2cnc[nH]2)OC2(CCC2)C1 N1(C(c2c(C)cc[nH]2)=O)CCCCC(NC(=O)Cc2nc[nH]n2)C1 c1(C(N2C(CNC(C(C)(CO)OC)=O)CCCC2)=O)cc2cccn2cn1 c1(C(=O)NCC2CCC(NC(=O)CN3CCOCC3)CC2)ccn2nnnc2c1 C1(CNC(CS(N)(=O)=O)=O)CC(F)(F)CN1C(c1csc(-c2cn[nH]c2)n1)=O CC(C)C(CNC(c1cnn(C2CCCC2)c1)=O)NC(C1CCCC1O)=O c1(N2CC(CC)OC(C)C2)nc(NC2CCCC2CO)c2ncsc2n1 C(=O)(C(C)CS(C)(=O)=O)N1C(CNC(=O)CC(F)(F)c2ccccc2)CC(OC)C1 C1(C(=O)NC(C(C)NC(=O)CCOCC2CCCO2)C)CCN(C)CC1 c1(OCC)ccc(CC(=O)NC2CCCCC2C(C)C)nc1 c1(C(N(C2CC(NC(c3c(NC)nccc3)=O)C2)C)=O)cc2ccc(C)cn2c1 O(NC(=O)CCC(C)C(=O)OC(C)(C)C)CC(N1CC(C)(CN=[N+]=[N-])C1)=O N1(C(C(CC)F)=O)CC(NC(c2cc(N3CCOCC3)ncn2)=O)CC(F)C1 c1(C(=O)NC2C(O)CCN(C(c3cn(C)nc3)=O)C2)ccn2c1CS(=O)(=O)CC2 c1(CCC(=O)N(C2CCN(C(c3n[nH]cc3C)=O)C2)CC)cncc(F)c1 c1(N2CC3C(C2)N3C(C2CN(C)C2)=O)ccc2nc(C)nc(S)c2c1.CO Cc1ccc(C(=O)NC2CN(C(C3CC(CF)C3)=O)CC2(C)C)c(F)c1F C1(NC(c2cccc(C#C)c2)=O)CCN(C(C23CC(C)(C2)OC3C)=O)CC(O)C1 c1(NC(CS)=O)ccc2c(c1)COC2.C(CC(=O)NC(C)CSCC)NC(=O)OC CN1CCOCCC1C(=O)NCC(O)C(=O)NCCCCCCC1CC1 c1(C(=O)NC2C3(CC(NC(=O)CCOC4CC4)C3)C2)nc2cccnc2s1 c1(C(C)C)ccc(C(=O)Nc2cc(CO)nn2C(C)(C)C)c(F)c1 CC(=O)C(C)(C)CC(=O)N1CCCC(F)(CNC(c2ccncc2F)=O)CC1 C1(C(=O)NC(C)CNC(=O)C(O)Cc2cnc[nH]2)CCN2CCCC2C1 C(=O)(C1Cc2ccccc21)NC(C1C(C)(C)N(C(=O)CNc2ccco2)CC1)=O C(=O)(CCS(=O)(=O)c1ccccc1)NC(CN(C)C(C1CC12CCC2)=O)(C)C c1(C(N2CCN(C(C(C)CN(C)C)=O)CC2C)=O)c[nH]c2cc(Cl)c(Cl)cc12 c1(OC)cc(N2CCN(Cc3ccnc(F)c3F)CC2)nc(C(F)(F)F)n1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(CCOCC#C)(C(=O)OC)CC1 C(CC(C)C)(C(=O)N1CC=CCO1)ONC(c1cccc(C)c1)=O N(C=CC(=O)C(F)(F)F)C(C1CC12CCN(Cc1c(SC)ccnc1)C2)=O Cc1cc(C(N2CCC(CN(C(=O)C(C)C(C)O)C)CC2)=O)nc(N(C)C)n1 C1(CNC(C(OC)OC)=O)CN(C(=O)CCc2ccon2)CC12CCC2 C1(C(N(CC#C)CC)=O)CCCN(Cc2ccc(CN(C)C)cc2)C1 N1(c2c(F)cnc(C)n2)C(CNC(=O)CCS(=O)(=O)N(C)C)CC2COCC12 C(=O)(CCCc1nc(-c2cccs2)no1)NC(C(C)OCC)C C1(CC=C)(C(=O)NCCCc2n[nH]c(C)n2)CCCN1C(=O)COC(C)=O C(C(C)C)(C(F)(F)F)NC(c1c(C)nc(CNC(=O)CCCF)o1)=O CCCC(C)(CCC)C(=O)N(CCNC(c1ccc2cc(C)oc2c1)=O)C1CC1 C1(CCC(=O)NC2(C(C)C)CC2)CCN(C(=O)C(O)CN(C)C)C1 NS(=O)(=O)C1(C(N2CC(CCCCNC(C3CC3F)=O)C2)=O)CC1 CCC(CCOC)C(=O)N1CCCCC1CCC(=O)NC1CCCN(O)C1=O Cc1ccc(CNC(=O)C(N2CCN(C(C3CCCOCC3)=O)CC2)C)cc1 N1(C(CC=CC(=O)NC2(c3cc[nH]n3)CC2)=O)CCC(Cc2ccccc2)C1 C=C(C)C(F)(F)CC(=O)NC1CCCN(C(=O)Cc2cscn2)C1 C1(NC(C(CCC)OCC)=O)CC12CCN(C(=O)C1=CCCOC1)CC2 c1(C(C)C)cccc(NC(=O)C(C)(C)C2CCN(C(c3ccccc3O)=O)C2)c1 C(=O)(CCc1ccc[nH]1)N(C(C(=O)N(C1CC(O)C1)C)C1CC1)C c1(C2C(C(=O)NCCN(C(C)C)C(C3CC(O)C3)=O)C2)ccccc1 c1(C(N2CC3CN(C(c4cc(C(N)=O)[nH]c4)=O)C3C2)=O)cc2ncccc2[nH]1 c1(C(=O)NC(CN(C(c2cnc(CC)[nH]2)=O)C)(C)C)ccc2sc(=N)[nH]c2c1 C(CC(=O)NCC)(C(C)OC(C)(C)C)NC(=O)Nc1c(CC)c[nH]n1 C(=O)(CCCCCNC(=O)CN1CCNC1=O)N1CC(CC(C)C)C1 N1(C(CCOC)=O)CCCC(C2CCCN(C(C3(CF)CCC3)=O)C2)C1 c1(C(=O)NC2C(NC(c3cc(C(C)=O)sc3)=O)CCC2)cc(C)nc(O)c1 c1(C(N2CCC(CC=C)(NC(=O)C3=CCCO3)C2)=O)cc(F)c(F)c(C#N)c1 N1(C(C2C(C)(CC)C2)=O)CC2(C1)CN(C(=O)C(=Cc1c[nH]cn1)F)C2 Cc1cc(C)c2cc(C(=O)NC(CNC(=O)CC3CCCO3)C(C)(C)C)[nH]c2c1 c1(C(=O)NCCCN(c2ncnn3cccc23)CC)ccc2c(c1)CCCO2 c1(C(=O)OC)nscc1NC(=O)C(=O)N(C)CCOC(C)=O c1(-n2ccc(CNC(=NC)NCC3CC=C(C)CC3)n2)ccc(Cl)cc1Cl CC(C)CC(C(=O)NC1CC(NC(=O)C(C)(C)c2ccn(C)n2)C1)C(N)=O c1(C(=O)NC(C(=O)NCc2cc(CC)[nH]n2)CC2CC2)cc(C#N)cn1C C1(CNC(c2cc(C)ncc2)=O)CN(C(=O)C(C)=C2CCC2)CCC1C(F)(F)F C(=O)(C(O)CC[S+](C)C)N1C(CCN(C(=O)C=C2CCN(C)CC2)C)CCCC1 C(=O)(CCC(=O)N1CCCCC1CCNC(C12COCC(C1)C2)=O)NCCC CN1C(=O)c2ccccc2C1CC(=O)N1CC(F)(CNC(=O)CCCF)C1 C1(c2cn(C(C)C(=O)N3CCCC3)nn2)CCCCCC1 C1(N(C(C2N(C(CCC)=O)CCC2)=O)C)CC2CC1N(C(c1cnc(S)[nH]1)=O)C2 C1(C#N)(C(=O)NCC(=O)Nc2cn(CC(C)C)nc2)CC(=O)C1 CCC(C)(O)C(=O)NC(C)C(C)NC(c1nn(-c2cccc(F)c2)cc1O)=O C1(NC(c2c(C)nc(CCC)s2)=O)CCC2CN(C(=O)CC(C)C3CC3)CC2C1 c1(C(=O)NC2C(NC(=O)CCF)COC2)n[nH]c2ccccc12 Cc1scc(C(=O)NCC(C)NC(c2cc(C#N)on2)=O)c1Br C12(C(=O)NC3CN(C(CCN(C)CC)=O)CC34CCC4)CCOC1CC(=O)NC2 C(C1CCCc2sc(C)nc21)NC(c1cccnc1)COC N1(C(C2C(C)C2)=O)CC2(CCC(CNC(=O)COCC3CC3)O2)C1 C1(O)(CC(=O)NCC=CCNC(C(c2ccccc2Cl)OC)=O)CCCCC1 N1(C(c2cn(CC=C)nc2)=O)CCC(CNC(C2CC(C)C2(C)C)=O)(OC)CC1 C=C(C)CC(C(=O)NCCC1(O)CCN(C(C2CCN(OC)CC2)=O)C1)OC N1(C(c2cc(CC)c(CC)o2)=O)CC2CCCC2(NC(=O)CN2CC3CC3C2)C1 Cc1cccc(F)c1CC(=O)NCC1CC1NC(C1CN2CCC1C2)=O N1(C(c2cc(CNc3ccnc(NC)n3)oc2)=O)CCC(C(=O)NC)C(O)C1 N1(C(=O)CCSc2ccccn2)CCC2CN(C(C3OCCCO3)=O)CCC2C1 C1(CNC(C(CC)C)=O)CC2(C1)CN(C(c1ccsc1-n1cnnn1)=O)C2 N1(C(C=CC)=O)CCN(C(c2cnc3n2CCS3)=O)C(CF)C1 c1(NC(C2CCC(CNC(C3CCCC3)=O)CC2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(c2ccc(C)[nH]2)=O)C(CNC(c2nccc(C(F)F)n2)=O)CC2COCC12 CCC1=C(C(=O)N(CC(C)NC(c2ccc(C(C)(C)C)nc2)=O)C)SCCO1 C#CCCCCC(=O)NC1CCN(C(=O)C(C)Oc2ccc(Br)c(C)c2)C1 C1(CC(=O)NCCC(=O)NC(CC)C)CN(C(=O)Cc2csc(C)c2)CC12CC2 C1(CN(C)C(C2CNC(=O)N2)=O)CCCCN1C(=O)CCSc1ccccn1 c1(NC(=O)NC(C(C)(C)OC)c2ccccc2)ccccc1OCC1CCCC1 C1(NC(c2c(CC)con2)=O)CC2CC1N(C(=O)C=Cc1cnn(C)c1C)C2 C1(NC(C(n2ccc(C)n2)C)=O)CC2(C1)CN(C(=O)C(CO)C(C)C)C2 CC(C)C(CNC(c1csc(C(F)(F)F)n1)=O)NC(c1ncoc1C1CCC1)=O CC1(C)C2CCC(NC(=O)CC3CCCN(NC(C4CC(O)(C#N)C4)=O)C3)C1C2 c1(CC(=O)N(CC(C)(C)CNC(=O)C(F)CC)CC)c(C)cccc1C CC1CCOCC1C(=O)N(CCCNC(=O)CC12CC(C1)C2)CCO c1(CNC(C=COCC)=O)nc2c(s1)CN(C(c1csc(NC(C)=O)n1)=O)CC2 Cc1cccc(C=CC(N2CCC(NC(c3oc(C(F)(F)F)nc3C)=O)C2)=O)c1 CCCC(C(=O)NC(C)CNC(=O)C(O)C(C)C)OCC C(=O)(CCC(F)(F)F)NCC(=O)NC(C(=O)OC)C1CC1 C1(N=c2ccc3c([nH]2)CCC3=O)(COC)CCN(C(=O)CSCC(N)=O)CC1 N1(C(c2cc(O)cc(F)c2)=O)CC2CCN(Cc3c(F)cccc3I)CC2C1 c1(CNC2CC(NC(=O)C=Cc3ccco3)C2)cccnc1O c1(C(=O)NCC2C(NC(=O)Cc3cncs3)CC2)cnc(O)s1 c1(NC(C(CC=C)C)c2nnnn2Cc2cccs2)ccc(OC)c(C)c1 O=C(Cc1nc(O)c2sccc2n1)NNc1ccc(F)c(F)c1 C1(CNC(C2N(C)CC2)=O)CCN(C(C2CCCOC2)=O)C1 c1(OC)cc(F)cc(C=CC(N2CCC(C#N)(NC(=O)CCC3CC3)C2)=O)c1 n1(CC(=O)NCCOC2CCN(C(C3(Cl)CC3)=O)C2)cnc(Br)c1 n1(CC(=O)NC2(CSC)CCC2)cc(CC(c2cc(C3CCOC3)[nH]n2)=O)nn1 C1(C)(NC(c2ccc(COC)o2)=O)CCN(C(=O)C(C)N(C)C)C1 c1(C(N2CCC(C(C)(C)NC(c3c(C)nsc3)=O)C2)=O)cc(F)cc(F)c1 Cc1ccc(CS(=O)(=O)NC2CCCC2C(=O)NN2CCC(O)C2)cc1 c1(C(=O)NCC2(CNC(C3(F)C(C)OCC3)=O)CC2)cccc2cc(Cl)ccc12 C1(CC(=O)NCC2(C(C)(C)O)CN(C(c3ccccc3)=O)C2)CCCOCC1 Cc1cc(C)c(C(N2CCN(C)CC2CNC(=O)C(O)P(C)(C)=O)=O)cc1C CC(C)(C)CCCC(=O)NCCCCCC(N1CCC2CCC(C1)S2)=O c1(OC)cccc(C(C)C(=O)NC(C2CC(NC(=O)C(C)(C)OC)C2)C)c1 CC(C)C(C#N)C(=O)NCCCC(C)NC(=O)CC(=O)Nc1ccc(F)cc1 C1(C(=O)NC(CCCC)CNC(=O)C(C)(C)F)CC2CCC(C1)N2C(C)C c1(C(=O)OC)ccc(CNC(=O)Cn2cc(CC3CC3)nn2)cn1 C1(CNC(C2COCC2C(F)(F)F)=O)CCCN(C(=O)CNS(=O)(=O)C2CC2)C1 Cc1ncc(C(N2CCCC(C(C)NC(=O)COCC(C)C)C2)=O)cc1C#N CC1=C(C(=O)NCC(C)(CO)NC(=O)Cc2cc(C)cc(F)c2)CCS1(=O)=O N1(C(c2c(CC)cns2)=O)CCCCC1C(C)NC(=O)C(F)=C1CCCC1 N1(C(c2nc(C)nn2C)=O)CCC(C)(C)C1CNC(C1COCCO1)=O N1(c2cc(Nc3c(-c4c(C)non4)noc3)nc(C(F)(F)F)n2)CCC2CCCCC12 C1(NC(c2cnn[nH]2)=O)CCN(C(=O)CCCc2cc(Cl)sc2Cl)CC1O CCCCC(CC)C(=O)N1CC(C)(C)CC1CC(=O)NCc1ncnn1C1CC1 C(=O)(C1CCc2nccn21)NCC(C(C)C)C(=O)NCCc1ccccn1 Cc1ccc(Cl)c(C(N2CC(NC(=O)C(F)C3CC3)CC3(CC3)C2)=O)c1O CC(CC(C)NC(=O)C(n1nnnc1C1CC1)C)N=c1[nH]nc(-c2ccon2)s1 c1(C(=O)NCC2(C(=O)NCC)CC2)c(C(F)(F)F)cnn1C C(C)(CO)(CN=c1[nH]c(=NC(C)c2cc(C)n[nH]2)c2c(F)cccc2[nH]1)OC c1(C(=O)NC2(C)CC(NC(c3c(CC)scc3)=O)C2)ccc2cnn(C)c2c1 C1(C(=O)NCCC2N(C(C(C)OCCC(C)C)=O)CCC2)CCOC(C(C)C)C1 Cc1[nH]nc(C(=O)NCC2(O)CN(C(=O)CC3C(CO)C3(F)F)C2)c1C(F)(F)F C=CC(C)(O)C(=O)N1CCC(O)(CNC(=O)Cc2cc(Cl)n(C)n2)C1 C1(NC(c2c(C(=O)OCC)scc2)=O)CC2CC(C1)N(C(=O)Cc1cnsc1)C2 C1(NC(c2c(CC)csc2)=O)CCCN(C(C2CCC3CC23)=O)C1C C#CCN(OC)C(=O)C(Cc1ccoc1)NC(c1csc(C#N)c1)=O c1(C(=O)NC(C2CCCCC2)CNC(C2C(C)C2)=O)cc([N+](=O)[O-])cnc1N N1(C(COc2ccc(C(C)C)cc2)=O)CCOc2cnc(Br)cc21 c1(C(N2CCCN(C(CCC(=C)C)=O)C(CO)C2)=O)cc(C)nc2c1CCCC2 Cn1nc([N+](=O)[O-])cc1C(=O)NCC1CN(C(=O)CC2CCOC2)CC12CC2 CC(C)CC(CC(=O)NCC1CCN(C(C2(C)CS(=O)(=O)C2)=O)CC1)CC(N)=O N1(C(c2ccccc2O)=O)CC(C)N(C(=O)C=C(C)c2cccs2)CC1C.CO S(=O)(=O)(c1ccc(Nc2ccc(C(N)=O)cc2Cl)cc1Cl)NCCSCC(C)C C1(C(=O)NCC(CNC(C2(F)CC2)=O)C(F)(F)F)CC2CC1CC2(F)F c1(OC)ccc(C(CC(=O)O)N(C=O)Cc2nc(C)cs2)cc1OC N1(C(C2CC(=C)C2)C(=O)N(c2ccccc2C)CC)CCc2n[nH]cc2C1 c1(OC)ccc(CO)cc1C(=O)NCCCC(C)NC(=O)C=CC1CCCO1 c1(SCC(N2CC(NC(C3CC4C(C)(C)C4C3)=O)C2)=O)ccc2c(c1)CCC2 O=C1NC2(CCN(C(C3C4CCN(C(C5(O)CCOC5)=O)CC34)=O)C2)CO1 c1(CC(=O)NCCOCCNC(Cc2cn(CC)nc2)=O)coc2ccccc12 c1(C(=O)NCCN(C(c2c(C)nc(C3CC3)o2)=O)C)cc(N)nc(Cl)c1 C1(C(=O)NC(CC=CC)C(=O)OCC)CC2(C1)CC1(CCC1)C2 C(=O)(N=c1[nH][nH]c2c1CN(c1ncc3ccsc3n1)C2)c1c(SC)ccs1 N1(C(COC(CC)C)=O)CCn2ncc(S(C)(=O)=NC(=O)C(C)CC)c2C1 C(=O)(C(CO)C(F)(F)F)NC(CCC#C)C(=O)NC1CC(O)C1OC c1(CC)cc(C(=O)N(C(C(=O)NC(CC)CCOC)C2CCCC2)C)ccn1 N1(CC=C)C2CCC1CN(C(c1cc(NC(=O)OC)c[nH]1)=O)C2 c1(C(=O)NCCC2CCN(C(C3CCCC3)=O)CC2)coc2c1CS(=O)(=O)C2 c1(N(CCCO)C)ccn2ncc(S(=O)(=O)NCc3ccncc3F)c2n1 C(C(C)(C)CN=[N+]=[N-])NC(C(C(C)C)NC(c1cn(CCC)nc1)=O)=O Cc1nn(C)c2sc(C(=O)NC3CCN(C(=O)Cn4cccnc4=O)C3C)cc12 C1(CCCC)CCC(NC(=O)C(N2CCC(C(=O)OC(C)(C)C)C2)=O)CC1 C(=O)(C(CNC(=O)CCOCCCOC)CC1CC1)NC(CC=CCC)(C)C c1(CC(=O)NCCC(O)CNC(C2(CO)CCCCC2)=O)cc(F)cc(F)c1 C1(NC(c2c(CC)cno2)=O)CCCC12CCN(C(=O)Cn1cc(C)cn1)CC2 c1(CC(=O)NC2CC(C)(NC(COCC#C)=O)C2)nn(C)c(=O)c2ccccc12 C(CC(C)(C)C)(C(=O)NCCc1ccnc(O)c1)NC(CC1C(C)C(=O)CC1)=O C1(NC(CCCC#CC)=O)COC2(CCN(C(=O)C(S(C)(=O)=O)C3CC3)CC2)C1 CCCCC(C(=O)N1CCC(C)C(N(C)C(C23CC(C)(C2)OC3C)=O)C1)C(C)C C1(C(=O)NCCCCNC(CCC(=C)C)=O)CCCC(=O)N1C c1(C(N2CC(CCC)N(C(C3CC3(F)F)=O)CC2)=O)cn2c(C)cccc2n1 C1(C(=O)NCC(CCC)C)CC(O)CN1C(=O)C(C(C)O)N(C)C C(=O)(CCCC(C)(C)C)NCCOCCN(C(=O)C=Cc1ccsc1C(F)(F)F)C c1(NC(C)=O)ccc(C=CC(N2CCCN(C(=O)C=CC(C)(C)C)CC2)=O)cc1 c1(C(N2CC(CCCNC(C3(SC)CC3)=O)OCC2)=O)cncc(Cl)c1C N1(Cc2ccc(S(C)(=O)=O)cc2F)CCC2(CC(O)CNC2=O)C1 C1(C)(CNC(c2nn(C)c(C3CC3)c2)=O)CCCN(C(C23CCC(C2)OC3)=O)C1 C1(NC(COCC)=O)COC2(CCN(C(c3cncc(OC)c3)=O)CC2)C1 N1(C(C)=O)CCCCC1COC(=O)N(CCN(C)C)CC1CC1 N1(C(Cc2cc(C)on2)=O)CCOC2(CCN(C(c3cc[nH]c3)=O)C2)C1 c1(C(=O)NCC23CC(NC(CSCC(C)C)=O)(C2)C3)csc2c(O)ccnc12 C(C)(CO)(C(=O)N1CCC(CCC(=O)N(C)CC2CCCC(C)C2)CC1)OC N1(C(c2ccc(-c3ccc(C)n3C)cc2)=O)CCC2(CC1)CC(F)CO2 CCCCCC(CCCCC)C(=O)NC1CCC(CNC(c2ccsn2)=O)CC1 N1(C(C2C(OC)CCC2)=O)CCC(C)C(CNC(C23CCC(CC2)C3)=O)C1 CCCCC(O)C(C)C(=O)NCC1CC2CN(C(=O)C(c3cnn(C)c3)=O)CC12 C1(N(C(c2cc(C)co2)=O)CC)CCCN(C(=O)CCC2CC(OC)C2)C1 c1(C(=O)NCC2=CCN(C(C3C(C)(CC)C3)=O)CC2)csc2ccc(C)cc12 N1(CCNC(c2ccc[nH]2)=O)CCN(C(c2cn3ccnc3s2)=O)CC12CCC2 C1(C(=O)NC2C3(CN(C(c4c(C)cns4)=O)C3)CCC2)CC(F)(F)CCC1(C)C C1(CNC(c2ccc(CC)o2)=O)(NC(=O)Cn2ccc(C)cc2=O)CCCCC1C Cc1cc(C)c(CCN=c2[nH]c(C(N3CCC(C(C)C)CC3)=O)cs2)c(C)c1 c1(C(=O)NC2(CO)CCCN(CC(COC)O)C2)sc2ccccc2c1Cl C1(NC(C(C2CCN(C(c3[nH]cc(C)c3)=O)C2)F)=O)CC2(CCOC2)C1 CC1(C(=O)NC2C3CN(c4nccc(S(C)(=O)=O)n4)CC23)COc2ccccc2O1 c1(NC(N2CCC(C)C(CCC(=O)O)C2)=O)cc2c(ccn2C)s1 n1(COCC)nnc(C(=O)NCCC(C)NC(c2cn(C)nc2C)=O)c1N C1(CNC(c2c(CC)n(CC)nc2)=O)CCCCN(C(=O)C(F)(F)C2CC2)C1 Cn1cc(C=CC(=O)NCC(C2CCN(C(c3ccccc3)=O)CC2)F)cn1 C=CC1(C(=O)Nc2cnc(F)nc2)CCN(C(c2nonc2C)=O)CC1 C(c1ccccc1OC)=CC(N1CCCC(NC(C(CC)SC)=O)CC1)=O C1(CNC(C(C)OCC)=O)CCCCC1C(=O)NC1(C(F)(F)F)CCC1 CCC(C#N)C(=O)NC1CC12CC(NC(=O)COCc1nnc(C)s1)C2 CN1CCn2[nH]c(=NC(=O)C3CCCCC3(C)C)cc2C1 C1(CCCC)CN(C(C2CN(C)CCO2)=O)CCN1C(c1cnc(S)nc1)=O Cc1cnc2n1CCCC2C(=O)NC12CCC(CC1)N(C(C1SCCC1C)=O)C2 C1(CC(NOCC(=O)OCC)=O)CCCN(C(C2CC(=O)N(OC)C2)=O)CC1 C1(C(N2CCC(F)(F)C2)=O)CCN(C(c2ccsc2)=O)C12CC2 c1(C(N2CCC(NC(CSC)=O)(CF)C2)=O)csc2c1CCC(C)C2 C1(C(N2CCCC(N(C)CCc3cc(Cl)cc(Cl)c3)C2)=O)CCc2nccn2C1 Cc1[nH]nc2ncnc(N3C4CCC3CN(C(=O)C(C)(C)n3cncn3)C4)c12 c1(C(C(=O)NC(CN(C(C(C)OC)=O)C)C)C2CCCC2)ccncc1 c1(C(N2CC3C(CNC(Cc4cnc(C)s4)=O)(C3)C2)=O)c([N+](=O)[O-])cnn1C c1(C(C)(F)F)cccc(NC(C2CCC(CNC(C3CCN3C)=O)C2)=O)c1 CC1(C)CCCCN(C(C2CCC(CNC(C3(C)CCOC3)=O)C2)=O)C1 N1(C(CC(CC(C)C)C)=O)CC2(CCOCC2)CC1CNC(C1(C(C)C)CC1)=O c1(C(=O)NC(CC=C)CNC(=O)C(C)CC(=O)OC)cc(C)cc2cccnc12 Cc1c(C(=O)N(CC(O)CN(C)C(C2(F)CC=CC2)=O)C)cncc1Br C1(C(=O)NC23C(CN(C(CCC#N)=O)C2)C3)OCC2COCCC12 C1(CNC(c2cc(C(C)C)[nH]n2)=O)N(C(=O)CCC2CC2)CCCC1(C)C C1(CNC(CS(C)(=O)=O)=O)CCC2(CN(C(=O)C(=Cc3ccccc3)C#N)C2)O1 C(CCCCCC(=O)NC1CCc2nncn2C1)NC(C(C(=C)C)(C)C)=O N1(C(c2c(C)oc(C(C)C)n2)=O)CCC2CN(C(=O)Cn3nccn3)CCC2C1 c1(C(=O)NCCC(C)(C)NC(CN(CCC)C)=O)cccc(C)c1F N1(C(c2ccc(SC)s2)=O)CCOC(CCNC(=O)C(N2CCC(C)C2)=O)C1 Cc1ccc(C(=O)NC2CN(C(=O)Cn3cc(C#N)cn3)CC2C)nc1 CC1=C(C(=O)NC(C)C(CO)NC(c2[nH]c(C)nc2C)=O)Cn2ncnc2N1C C1(CNC(CSC)=O)CCCN1C(=O)C(C)(F)c1ccccc1 c1(C(N2C(CNC(c3ccc(Cl)c(O)c3)=O)CCCC2)=O)cc([N+](=O)[O-])ccn1 CCCC(CNC(=O)C(F)C(C)CNC(C1CNC(=O)N1)=O)CCC C1(C(=O)NC(CCCC)C)C(C)OCCN1C(=O)Cc1ccc(F)nc1 CCCCC(CNC(C1C=CC=CC=C1)=O)NC(c1cccc(C2CC2)c1)=O c1(OC)ccc2nc(CNC(=O)C(N3CCCC3c3ccccc3)=O)ccc2c1Br c1(C(=O)NCCCOCCN(C(c2n(C=C)nnc2)=O)C)cccc(F)c1NC C1(CN(C(C2(CC=C)CCCC2)=O)C)CN(C(c2cc(Cl)n(C)n2)=O)CCO1 c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)(F)F)cccc2nc(C)nn12 N1(C(c2n(C)c(O)nc2)=O)CCC2CCN(C(=O)CCC=CBr)C2C1 Cc1nn(C)cc1C(=O)N(C(C)CCCNC(=O)COC1(C)CCCC1)C1CC1 c1(CN2CC(C#N)C(NCc3ccc(C(=O)O)s3)C2)cc2ccccc2o1 Cc1cnc(CNC(=O)Cc2cccc(C)n2)c(C)c1 C(=O)(CCC(C)(C)C)N(CCC(N1CC(N(C)C)C1)=O)C1CC1 Cc1c(S(=O)(=O)NC2CC(O)CN(C(=O)C(F)(F)F)C2)oc2ccc(F)cc12 CC(C)CCN=C(NCC1(C)CCCO1)NC1CCCC(F)(F)C1 c1(C(=O)NCC(CNC(C2(C)CCCC2(F)F)=O)F)nc[nH]c2ncnc1-2 CCCCS(=O)(=O)NCC(=O)NCC1(F)CC(NC(=O)CC(=O)OC)C1 c1(C(=O)NC(C(=O)NOCC=CCl)C2CCOC2)cnc(S)nc1 C1(NC(=O)Cc2ccco2)(CF)CCN(C(C2CCC2c2nc[nH]n2)=O)C1 C1(NC(C=CC)=O)CCC2CN(C(c3ccc(OC(F)(F)F)cn3)=O)CC2C1 CC(C)(COCCO)C(=O)N1CCC(n2cc(COc3cnc(S)[nH]3)nn2)C1 Cc1cc(F)c2cc(C(=O)NC3CCN(C(C4(CO)CC4)=O)C(C)C3)[nH]c2c1 C1(CCOC)CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)CCc1cnn(C)c1 c1(OCCC)ccccc1C(N1CC(NC(C2CC(C)CCO2)=O)C(C)C1)=O C1(Cn2cc(C3(F)CN(C(Cc4cnc(C)o4)=O)C3)nn2)CCS(=O)(=O)C1 CCC1=NOC(CNC(C2COCCC2CO)=O)C1.c1(C(=O)N)cnc(C2CC2)o1 C=CCC(CC)C(=O)N1CCCC(C)(CNC(c2ccc(CCN(C)C)cc2)=O)C1 Cc1nccc(COC(c2ccc(C3(O)CCCCC3)cc2)=O)n1 N1(CC)CCOCC1C(N1CC(C(=O)N(C)Cc2ccsc2)(SC)C1)=O C1(NC(c2c(C)cn(C(C)C)c2)=O)CCN(C(=O)CSc2nncn2C)CC1C C1(CN2C(C(=O)Nc3c(OC)ccc(F)c3)CCC2C)CCCC2CCCCC12 c1(CNC(=O)NCCC23CC(C)(OC2)C3)ccc(Cl)c(Br)c1F N1(Cc2ccc(C)nc2)CCC(C#N)(NC(=O)C(N)=O)CC1 N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(c2[nH]nnc2C2CCOC2)=O)C(C)C1 N1(CCNC(c2scc(C)c2Cl)=O)CCCN(C(=O)CCCC2CCCC2)CC1 CC1CCOCC1C(N1CCC1CC(=O)NCCN1CCOCC1C)=O O=C(CCCCC1CC1)NCCCN1CCN(C(c2ccc(Cl)o2)=O)CC1 C1(NC(C(c2cccc(F)c2)(C)C)=O)CCCCC1NC(C1CNC(=O)C1)=O c1(C(=O)NCC=CCNC(C(C(CC)C)C)=O)ccc(F)c(Cl)c1N C1(C(N2CC3(C2)CC(=O)N3)=O)CCCOCC1.C1(C(=O)OC)CC(n2cnnc2)C1 C(CC1CCCCC1)(C(=O)OC)ONC(C1CCNC1=O)=O.C(C(=O)O)OCCC C1(NC(C(C)SC)=O)CC2(CCN(c3cc(C)c(C(F)(F)F)cn3)C2)C1 C1(N(C)C(C2(C#N)CC2(C)C)=O)CN(C(=O)CCC(F)(F)F)CC1(C)C CCC(CCC(=O)NCC1CC(NC(=O)CC(=O)N(C)C)CO1)OC c1(CCC(N2CCCC(N(C)C(C3CCNC(=O)C3)=O)C2)=O)cccc(Cl)c1Cl N1(C(Cc2nc(CC)sc2)=O)CCC(NC(=O)C(O)COC)C12CC2 c1(C(=O)NCC2(C(=O)OC)CCCO2)cccc(-n2[nH]nnc2=N)c1 C1(C(N)=O)(CNC(CC2(C)CC2)=O)CN(C(C2COC(=O)N2)=O)C1 C#CCC(C)(C)C(=O)N1CC(NC(C2(n3cnnn3)CC2)=O)C(C)C1 c1(C(=O)NC2CN(C(C(CC)(C)F)=O)CC2SC)cnn2cccnc12 C1(CNC(C(CCOC)C)=O)CN(C)CCN1C(=O)CSc1ccc(C#N)cc1 N1(c2cc(OC)ncn2)CC2C(C1C(=O)Nc1cccc(O)c1F)C2(C)C N1(C(=O)C=CC=O)CCC(O)C(N(C(=O)CC2CC3(CC3)C2)C)C1.CNC C1(N(C(C(C(=O)OC)C)=O)C)CCCN(C(c2cnn(CCF)c2)=O)CC1 C(=O)(C(=O)N=S(C)(C)=O)NCCOCCCN(C(c1c(Cl)cc(C)s1)=O)C Cc1cc(C(N2CCCC(CCNC(C34CC(C)C3C4)=O)C2)=O)nn1C c1(OC)csc(C(=O)N(C)CC2CN(C(=O)CC3CC3C(C)O)C2)c1OC N1(C(C(CCSC)O)=O)CC2(CCC(NC(=O)CCCC(C)O)CC2)C1 C1(C(N2C(C(C)C)C(C)(C)C2)=O)CNC(=O)CN1C(=O)CC1CCC1 C1(C(=O)NC(C2(OC)CCC2)C)CC=CCN1C(=O)Cc1cc(C)n(C)n1 CC1(CC(=O)NC(C)(CNC(=O)CC2COCCO2)CO)OCCO1 c1(CC)ccc(CNC(=O)C(=O)N(CC(F)CC)CC)nc1 Cc1ccccc1CCC(=O)NCCCCCCNC(C1CC(C#N)C1)=O c1(CC)[nH]nc(Cl)c1C(=O)NC1CCCCC1NC(=O)C(c1ccccc1)C CCCCC(O)CC(=O)N1CCN(C(c2cn(C)c(C)cc2=O)=O)CC1CCO C1(CNC(CC2(OC)CCC2)=O)CCN(C(=O)CC2CCCC2C)C1(C)C C1(C(C(=O)NCC2(OC)CCN(C(c3cc(C)on3)=O)C2)O)CCCCCCC1 C(=O)(NNc1c(F)cc(F)cc1I)C1CC(NCc2scc(C(=O)O)n2)C12CCC2 c1(N(C(C2(C(=O)O)C(C)(C)C2)=O)CC2CC2)nc2c(s1)CC(F)(F)CC2 N1(C(COCCCCC)=O)CCOC(C(C)NC(=O)CC2CCC(OC)CC2)C1 CCCCC(=O)NCC(=O)N(CCCN(C)C(c1c[nH]nc1CC)=O)C N1(C(C(C2CCOC2)OC)=O)CC(NC(C2CCCC2)=O)C2(CCOCC2)C1 C1(N(C(c2c(OC)csc2)=O)C)CCN(C(c2cc(CC(C)C)on2)=O)CC1C N1(C(COCCC#C)=O)CC(NC(=O)CNS(=O)(=O)N(C)C)CC12CCOC2 C12(CNC(c3ccc(C(C)=O)[nH]3)=O)CC(CCO1)N(C(=O)C(C)O)C2 c1(C(N2CC=CC(NC(c3c(C)oc(C4CC4)n3)=O)C2)=O)nnn2c1CSCC2 Cc1ccc(O)c(C(=O)NCC2(F)CCN(C(C3NC(=O)OC3C)=O)CC2)c1 N1(C(C(COC)C)=O)CC(NC(c2cncc(N(C)C)c2)=O)C(C(F)F)C1 C1(C(=O)NC(C2CCOC2)CNC(c2ccn(C)n2)=O)CCC2(CC1)CC2(F)F C(CCCCCCCO)=CC(N1CC(C)C(CNC(C2(F)CC3(CCC3)C2)=O)C1)=O C(=O)(C1=Cc2cc(Br)ccc2OC1)NC1CCC(CNC(CNC=O)=O)C1 C(=O)(C1=CCC(C)(C)CC1)NC1CCC(C)N(C(=O)CCc2cn(C)nn2)C1 C#Cc1ccc(C(=O)NC(C(=O)O)C(O)Cc2ccccc2)nc1 c1(NC2CN(C(CCC(C)SC)=O)C(C)CC2)ncnc2c1ncn2C C1(C2CN(C(C3CCCOC3C=C)=O)C2)(NC(CSCC=C)=O)CC1 c1(NC(C(C2CC2CC)N(C)Cc2ccccc2C(F)(F)F)=O)ccc(Cl)cc1 C#CCC(C)(C(=O)NCCN(C)C(C)C)NC(=O)Cc1cn(CC)cn1 N1(C(c2c(C)nn[nH]2)C(=O)NCCOC)CCN2CCCCC2C1 Cc1cc(C(N2CC=C(C(=O)NCC3CC34CCOC4)C2)=O)nc(O)n1 C(c1cccc(F)c1)=CC(=O)NCC1CN(C(=O)CCCF)CCO1 N1(CC)C(=O)CCC1CC(=O)NCC=CCN(C(C1C2(CC2)C12CC2)=O)C1CC1 C1(C(=O)NC(C)C#N)CC(O)CCN1C(=O)C(N)=O C1(C(=O)NCC(C)(O)C2CCCC2)CN(C(=O)CC2CC(=O)C2)CCO1 c1(N(C2(C#N)CCNC2)C(=O)CCNc2cnc(Cl)c(I)c2)cccc(Cl)c1O c1(OC)ccc(S(=O)(=O)NC2CCC(C(=O)NC3COCC3O)OC2)c(F)c1 C1(CC(=O)NC(C2CN(C(=O)CCCC3CCC3)C2)CO)NC(=O)NC1=O c1(N(C(=O)C=C2CCOCC2)CCOC)ccc(C)cc1 N=c1[nH]cc([N+](=O)[O-])cc1C(=O)NCC1(NC(c2cc(Br)no2)=O)CC1 C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)CCc2csc(C)n2)CC1C N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CC(C)(C)OC)C2CCCCC12 CC1CCN(C(=O)CCNS(C)(=O)=O)CC1CNC(C1CC(=O)NC1(C)C)=O c1(CNC(C(COC)C)=O)cc(C(=O)NCc2cc[nH]c2C(N)=O)nn1C CC1CCN(C(c2cncs2)=O)C(CNC(C23CC(F)(C2)C3)=O)C1 C1(CNC(c2n(C)ncc2)=O)COC2(COCCN(C(C3(C)CCC3)=O)C2)C1 C(=O)(C(CCF)NC(=O)CCOC(C)C)NC1(CSC)CC1 N1(C(C2(CC(C)=O)CC2)=O)CC=C(C(=O)NOCCN(C)C)C1 C1(NC(C(CC#C)C)=O)C(C)(C)C(NC(c2cc3oc(C)cc3[nH]2)=O)C1(C)C C(=O)(C1=CCC2(COC2)OC1)NCCN(C(c1cc(CN(C)C)on1)=O)C1CC1 C(=O)(C1=CC2CCCCCC12)NCCC(C)N(C(C1(OCC)CC1)=O)C Cc1[nH]c(C#N)cc1C(=O)NCCCNC(=O)C1=CC(C)CC1 N1(C(C2C3(CCN(C(CC4(COC)CC4)=O)C3)C2)=O)CCc2ccncc21 c1(CC)ccc2c(c1)CN(C(C1CN(Cc3ccc(O)c(Br)c3)CCC1O)=O)C2 C(=O)(C(C)(C)C(O)CC)N1CC(CNC(c2ccc(OCCC)cc2)=O)OCC1 N1(C(CCCCOC)=O)CC(NC(c2ccc(Cl)cc2N)=O)C2(CC2)C1 C1(NC(C(CC#C)NC(=O)C(=Cc2cn[nH]c2)C)=O)CC2(CCC2)C1OC C1(CN(C)C(c2ccc(CO)cc2)=O)CCCCN1C(C1CSCN1C)=O C1(CC(=O)N(C2CCCN(C(C3CN(C(C)=O)C3)=O)C2)CCC)CCN(C)CC1 C1(NC(C2(CCCC)CCOC2)=O)CCC(NC(=O)CC2(C)CCCC2)CC1 c1(OC)ccc2cc1C(=O)N2.c1(CN(C)C)nc(C(C)C)ns1 C1(NC(c2c(C)csn2)=O)CN(C(=O)CC2CCCCN2C)CC1N=[N+]=[N-] c1(C(=O)NC(CC=C)CNC(=O)C=CCN(C)CC)ccc(C2CC2)cc1 C1(C(N(CC(C)CNC(C2COCC2n2ccnc2)=O)C)=O)CC(S(C)(=O)=O)C1 Cc1nc2cc(C(=O)NC3(C)CN(C(C4(C)CCCO4)=O)C3)ccc2n1C C1(C(N(CC(c2ccccc2)(C)F)C)=O)CCCC12CNC2 n1(CC(=O)Nc2ccc(NC(C(C(C)SC)O)=O)c(C)c2)ncc2ncccc12 C1(C(=O)NC(CNC(C(CC)NC2CCCC2)=O)CO)CCn2c(O)nnc2C1 C1(C(=O)NCCC2CCN(C(C(C)(C)c3cnsc3)=O)C2)CCCC12CC2 C(=O)(CCC(C(=O)OC)NC(=O)C(C1COC1)N(CC(F)Cl)C)OC C1(C(N2CCN(CC(C)C)CC2)=O)CC(F)CCN1C(=O)C(C)S(C)(=O)=O C#CCC(CC(=O)NCC1(CO)CCCCC1)NC(=O)C(C)C1CCC1 c1(C(C(=O)NCC)N(CCC(=O)OC(C)(C)C)C)cccc(C)c1F C1(C(=O)NC(CCCCNC(C(CCOC)(C)C)=O)CO)CC2CCCC(C1)C2 N1(C(C2(CC(=O)NC(c3ccoc3)=O)CCC2)=O)CC(O)(COCC)C1 C1(C(=O)NC2(C(=O)NCC3C(C)C3C)CC2)C2CCCCCC12 c1(C(N2CCN(C(=O)C=Cc3cccs3)C(CF)C2)=O)cccc2nncn12 N1(C(C=C(C)C(F)F)=O)CCC(NC(=O)C(O)CC(F)F)C(C)(C)C1 C(=O)(C1=NOC(CNC(c2sccc2CO)=O)C1)NC(CCC)CO CC(C)CC(O)CC(=O)N1CC(CCC(=O)NOCc2cccc(F)c2)C1CO c1(C(=O)OCC2CC(OC)C2)ccc(Cl)c(Cl)c1 c1(C(=O)NCCc2c(C)ccs2)ccc(-c2ccco2)cc1 C1(CNC(c2ccnc3ccnn23)=O)CC2CCC(C1)N2c1nc(Cl)ncc1F c1(C(=O)OCc2ccc(C)s2)c[nH]nc1S(N)(=O)=O N1(C(c2c(CC)c[nH]n2)=O)CCC(CC(=O)NCC(C2CCOCC2)O)C1(C)C C=CCC(F)(F)C(=O)NC1CCCC(N(C(=O)CNS(N)(=O)=O)C)C1 Cc1cc(N)c(C(N2CCOCC2CCNC(C23CC(C2)C(C)O3)=O)=O)nc1C C12(C(=O)Nc3c(C(C)=O)ccnc3)CCCC1(F)CNC2 C(=O)(C(CO)NC(=O)C(C)C1CC1)N1C(C(C)C)CC1 C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(c2ccc(N)cc2O)=O)C1(C)C C1(CC(=O)NC2(CN(C)C(C3C4COCC34)=O)CC2)CCCC2(CCC2)O1 C1(C(=O)NC2CCN(CCCO)C2)CC2CCC1N2C(c1cnc(O)c(F)c1)=O N1(C(c2ccsc2Br)=O)CCN(C(c2ccccc2)=O)C(CO)C1 CC1(C)CCCC(CN2CCCC2)O1.c12noc(=O)n1CCOCC2.c12ccc(cc1)o2 CCC(C)(C)C(O)C(=O)N1CCC2(NC(=O)COC3CCCCC3)CCCC12 C(c1cnn(C)c1C)=CC(=O)NC1CC(CCNC(C2ON=C(CC)C2)=O)C1 C1(N(C)C(C2CSCC(=O)N2)=O)CN(C(=O)C(Cl)=CCl)CC1(C)C Nc1cccc(C(N2CCCC(CCCCNC(C3CCCOC3)=O)C2)=O)n1 c1(C(=O)Nc2n(CC)nc(C)c2)cnn2cccc(-c3ccsc3)c12 N1(CC2(NC(=O)NC3CCCC(C(C)(C)C)C3)CCOC2)CCS(=O)(=O)CC1 C1(NC(C)=O)CCCC(CNC(=O)C(=O)NCC(F)F)C1 C(C)(CC(=O)NCCC1CCN(C(=O)CCC2CC2)CC1)(C(F)F)N(C)C C1(C(=O)NC2CN(C(=O)CC3(O)CC3)CC2O)CCC2(CCC2)CC1 Cc1ccc(C(F)(F)C(=O)NC(C)C(CO)NC(=O)C=Cc2cn(C)cn2)cc1 c1(CCNC(C(CCC)C)CO)ncc(C)cc1S(=O)(=O)N1CCSC(C)(C)C1 N1(C(C(C)CN2CCOCC2)=O)CC(CNC(=O)CNC(N)=O)CC(C)(C)C1 c1(C(N2CCCC(OC)C2)=O)cc2c(s1)CCN(CC1CCC(C)O1)C2 C1(NC(=O)CSc2nc[nH]n2)CC(CNC(c2ccccc2CO)=O)C12CCC2 C=C1CC(C(=O)NC2CCCC2NC(C2(C(C)C)CCC2)=O)(C(F)F)C1 Cc1cc(CC(N2CCN(C(=O)CCN3CCN(C)CC3)CC2)=O)c(C)n1C N1(S(CC2(NC(C)=O)CCOCC2)(=O)=O)CCc2c(ncn2C)C1C N1(C(C(c2ccco2)NC(=O)CCO)=O)CC([N+](=O)[O-])C1 CC(C)CC(C)(C)C(=O)N1CCC(O)(CNC(C2(O)CCSC2)=O)CC1 c1(NC(C2CCCN2Cc2ccc(-c3ccccc3)s2)=O)ccc(Cl)c(Cl)c1F N1(C(C(C#C)(C)C)=O)CCC(C(=O)NCC2(CC)CCCO2)C(O)C1 c1(-c2n(CC(CCC)C)ccn2)ccc(C)cc1.c1(S)ccccc1 C1(C(=O)NCC2=CCN(C(CC3(C=C)CC3)=O)CC2)CCc2n[nH]cc2C1C C1(CNC(C2CC(O)CN2CC2(C)SCCCS2)=O)C2CCCCC12 C1(NC(N2CCCC2CC2CC2)=O)CC(=O)N(C(C2CC2)C2CC2)C1 N1(C(C(C)(C)O)=O)CCC2(C1)CN(C(C1CC3CC(O)CC(C1)C3)=O)CCO2 C1(C(C)NC(=O)OC2CCOC2)CCN(C(=O)N(C)CCO)CC1.C1(C)CC1 C1(CNC(c2c(C)cc(C)[nH]2)=O)CN(C)CCN1C(=O)CCNC(C1CCC1)=O c1(C(=O)NCC2CCN(C(C(CC(=C)C)OC)=O)C2)cc(S(C)(=O)=O)ccc1C c1(CN(C(C(C2CC2c2ccccc2)NC)=O)CCO)cc2sccc2s1 N1(C(C(C)(O)C2CCC2)=O)CCC2(CCCN(C(C3(O)CCSC3)=O)C2)C1 c1(C(=O)NCC(CC)NC(=O)CC2CCC(F)(F)CO2)cn2cc(C)sc2n1 C1(NC(c2nc(C)n(C)c2C)=O)CN(C(c2cc(O)ncn2)=O)C2(CCC2)C1 N1(C(C(=Cc2cccs2)C)=O)CC2CN(C(c3cc(C)cc(C)c3N)=O)CC2C1 c1(C(=O)NC(CC(C)C)C(=O)OC(C)C)ccc2c(C(=O)NC3CC3)n[nH]c2c1 c1(OC)ccc(C(N2CC3(CCN3C(c3ccsc3OC)=O)C2)=O)cc1[N+](=O)[O-] N12CCc3c(ccnc3C1=O)C2.N1(C(CC)=O)CCC(C(=O)OC)C12CCC2 C1(C(=O)NCC2N(C(COCC(=O)OCC)=O)CCC2)CC2(C1)CC2F N1(CC(=O)OC(C)(C)C)CCC2(CCCCC2C(=O)NSc2cccc(C(=O)O)n2)C1 C1(C)(CNC(COCCOC)=O)CCN(C(=O)C=CC(N2CCOCC2)=O)C1 C(=O)(CC(O)CNC(=O)Cn1ncnn1)NCCCNC(=O)NC c1(C(=O)NC(CC)CNC(=O)CCOC)ccc(N)c([N+](=O)[O-])c1 N12CC3C(C3C1)CC2=O.n1(CC)ccc(C(N2CC=CCC2)=O)n1 CC(C)CC(C(=O)N(CCCO)CCCO)ONC(c1cnn(C)c1)=O CC1(C)OC(=O)CC1C(=O)NC1(C)CN(C(c2cnc(CSCC)nc2O)=O)C1 C1(OCC)COCCC1CC(=O)NCC(C(C)(C)C)NC(=O)CCC=C(C)C Cc1cn2c(=O)c(C(=O)NCC(C)(O)CNC(=O)Cc3cn(C)nn3)cnc2s1 CCC(CC(C)C)C(=O)N1CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)CC1C(C)C C#CC1(O)CN(C(=O)CN(C2CC(C#N)C2)C(=O)CN2CCCC2=O)C1 c1(C(CC)NC(C(CC(=C)Cl)n2cc(CCOC)nn2)=O)n[nH]c2ccccc12 C(=O)(C(O)C1=CCCCC1)NCC12CN(C(C3(CCC)CC3)=O)CC(F)(C1)C2 c1(C(=O)NC(C)CNC(c2nc(Cl)ccc2F)=O)cn2c(n1)CCCC2 C1(OC)CCN(C(c2cccnc2CNC(C2CC(C(=O)OC)C2)=O)=O)CC1 c1(N2CCN(C3CN(C(C4C(C)C4)=O)C3)CC2)nc2c(cc1C#N)C(=O)CCC2 CCS(=O)(=O)CC(=O)NCC(F)CNC(=O)CCNC(c1ccc(OC)cc1)=O c1(CCC(=O)NC2C(NC(c3cnc(CN(C)C)[nH]3)=O)CC2)ccc(Cl)cc1 C(=O)(C1=NOC(C2(O)COC2)C1)N1CCC(OC(COC)(C)C)CC1 Cc1cc(C(=O)NCC2CC(NC(C3CCC4(CC4)C3)=O)C2)c2sc(=N)[nH]c2n1 Cc1nn(C)c(C)c1C(=O)C(=O)N(C)CCOCCNC(=O)CCc1ccon1 C1(C(=O)NC2CN(CC(=O)Nc3ccc(OC)cc3)C(C)C2)CCCCNC1=O N1(C(=O)C#CC2CCOC2)CCC2(CCN(C(=O)C(O)CC(F)(F)F)C2)C1 c1(C(=O)NCC2C(C)CCN2C(c2cccs2)=O)cc(F)ccc1Cl c1(OC)cc(F)c(C(=O)NCC2(Cl)CC23CCC3)cc1Cl C(=O)(C#CC1CCOC1)NCC(C(=O)N1CCC(C(C)C)C1)(C)C Cc1cnc(N2CCN(C)CC2CNC(C2(C)CC2)=O)nc1C CC(C#N)CCC(=O)OCC(c1cc(Cl)ccc1Br)=O Cc1cccc(CCC(=O)NC(C(C)NC(=O)CCc2cncn2C)C(C)C)c1 C1(CC(=O)Nc2c(OCC)nccn2)CN(C(c2conc2C)=O)C(C)(C)C1 C1(NC2CCN(C(c3n(CCOC)ncc3)=O)CC2C)CC2(CCOCC2)C1 N1(C(CCCOc2c(C)cccc2)=O)CCCCC(NC(c2scnc2C)=O)C1 c1(CCC(c2cnc(C(N)=O)s2)N)ccc(Cl)c(Cl)c1.C1CC(=O)N1 c1(C(=O)NC(CCCNC(Cc2n[nH]c(=NC)s2)=O)C)cc2cc[nH]c(=O)c2s1 N(C(=NCCC(C)C)NC1CCC(C(C)C)C1)CC1(OC)CCCCC1 C1(C(=O)NCC2C(NC(CSCCCC)=O)CCCC2)CC2(CCC2OC)C1 C(C)(CC(C)(C)C)(c1n(CCC)nnn1)NC1CC(c2ccc(F)cc2)C1 O=C1Cc2c(NCC3CN(C(c4c(O)ccc(Br)c4O)=O)CCO3)ncnc2N1 C(CNC(c1sccc1C#N)=O)(CC(=O)NC1CC(C(C)O)C1)OC N1(CC(=O)NC2CCOC(C(N3CCC4CC34)=O)C2)C(=O)CCC1=O C(C)(C)(C(C)CC(=O)N1CCC2(CC1)N=N2)NC(c1c(C)[nH]cc1)=O CC(C)C(C)(CNC(C1CCC(CCO)CC1)=O)NC(c1csc(C(F)F)c1)=O N1(C(Cc2ccn(C)n2)=O)CCCC(C2CCN(C(c3cocn3)=O)CC2)C1 CC(CCCCNC(c1cc(C(N)=O)cs1)=O)NC(c1cn(C2CCC2)nn1)=O N1(C(CC(CC)C)=O)CC(C)(C)OCC1CNC(c1ccc2cc[nH]c2n1)=O CC1CC=C(C(=O)NC(CC(=O)N(C2CCCCC2)C2CC2)C(F)(F)F)CC1 c1(CC)ccc(C(N2CCOC(CC(=O)NC3CCOCC3C)C2)=O)cc1 c1(C(=O)NC(C)C(C)NC(c2cnc(O)o2)=O)cc(Cl)cc2ccccc12 c1(OC)ccc(NC(N2CCN(Cc3[nH]ccc3C)CC2)=O)c2ncccc12 CCCC(C(O)C(=O)N(CCN1CC=CC1)CC)NC(=O)C1=CCCC1C c1(CC(C)NC(CC)Cc2ccc(Br)cc2)c[nH]c2ccccc12 C1CCC(CNC(C2CCCOCC2)c2nnnn2CCc2ccccc2)CC1 C1(C(=O)NCC(CNC(c2cn(C)nn2)=O)(C)O)CCc2ncnn2C1 C=C(F)CN=c1[nH]c2cc(Cl)c(S(=O)(=O)N3CC4(CO)CCC3CC4)cc2s1 C1(N(C)C(c2ccn(CCF)n2)=O)CN(C(=O)Cc2csc(S)n2)CC1F c1(COC)nc(CC(=O)NCC2COCC2NC(=O)C(c2ccnn2C)O)cs1 c1(CCCC(=O)NCCCCNC(C2CC2CF)=O)ccc(C(F)(F)F)cc1 c1(C2C(=O)N2C)ccc(OC(F)F)cc1.C(CC#N)NCCOC(F)F N1(C(CCC(=O)OC)=O)CCOC2(CCC(NC(=O)CC3CC3C)CC2)C1 N1(C(CN(C)C)=O)CCCC(C2CN(Cc3cc(Cl)ccc3[N+](=O)[O-])C2)C1 c1(C(N2C(CCNC(C=NOC)=O)CSCC2)=O)cc(Cl)c(O)cc1C C(=O)(C1=CCCC1C)NC1CCC(CC(=O)N(C2(CCO)CC2)C)C1 C1(CCC(=O)OCC(c2ncc(-c3ccccc3)o2)=O)CCCCO1 N1(C(C2C(CC)OCC2)=O)CCC(NC(=O)C=C2CN3CCC2CC3)C(F)C1 n1(CC)cnc2c(NCC3(C)CCCC3O)nc(N3CCCC4(CCC4)C3)nc12 c1(CC(N2CCC(C(N3CC(OC)C(C)(C)C3)=O)C2)=O)cnc2ccccn12 CS(C)(=O)=NC(=O)C(=O)NC1(C)CC(NC(c2ccc(Cl)c(Cl)c2)=O)C1 c1(SC)cc(C(N2CCCC(NC(=O)CC3COC4CC3C4)C2C)=O)ccc1N N1(C(C2C3CN(C(c4c(C)[nH]c(C#N)c4)=O)C2C3)=O)CC2(C1)OC(=O)NC2C C1(C(=O)NC(c2ccc(Cl)cc2)C(=O)NCC(CSC)OC)CC(=O)NC(=O)N1 CN1CC2CC1CN(C(C1CN(C(c3ccc(=O)n(C)c3)=O)C(C)(C)C1)=O)C2 C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NCCN2CCCC2=O)CCCC1 N1(C(CC(C)OC)=O)CCC2(CC1)CCN(C(C1(Cl)CC1)=O)CC2 C#Cc1ccc(C(=O)NCC=CCNC(c2c(Cl)nn(C)c2C)=O)cc1Cl N1(C(CCS(C)=O)=O)CC2CCN(C(=O)C(F)C(C)(F)F)CC12 Cc1cn2ccnc(C(N3CCCC3CN(C)C(C3CCC(=O)N3)=O)=O)c2n1 N1(C(CCCN(C(C)C)C)=O)CCC(C)C1C(=O)NCCCCCO c1(CC)nc(C)oc1C(=O)NCC1(C)CCCN1C(C1CN(C)CCO1)=O CCCC(CCNC(C1(N(C)C(C2CCCN2C)=O)CC1)=O)C1CC1 N1(C(C(C)C)=O)CCC2(CCCC2NC(c2cc(CF)on2)=O)CC1 C1(CC(=O)NCCN2CCN(C(=O)CN3CCS(=O)CC3)CC2)CCS(=O)(=O)C1 N1(c2n3ccnc(C)c3nn2)CC2(CN(C(=O)OC(C)(C)C)CC(C)(C)O2)C1 c1(C(N(C(CNC(C2CC(C)(C)O2)=O)C2CC2)C)=O)ccn2ccnc2c1 N#Cc1c(Cl)cc(C(N2CC(CNC(=O)CN3CCOCC3)C2)=O)cc1Cl C1(CNC(=O)C=CCO)CC12CCN(C(c1cc(Cl)c(Cl)s1)=O)CC2 C12(C(=O)NCC3(O)CN(C(C(C)C4CCC4)=O)C3)C3C4C1C1C2C3C41C c1(C(=O)NCC(CNC(C(C)(O)C2CC2)=O)O)cnc(O)cc1O C(=O)(C1Cc2c(Cl)cccc21)N1CC(OC)(CNC(C2(C)CCC(C)C2)=O)C1 c1(OC)cccc(C)c1C(=O)NCC1CCCCN1C(=O)Cc1cscn1 C1(NC(=O)CCCc2cnn[nH]2)CN(C(=O)C=CI)CC2(CC2)C1 C#Cc1cc(NC(=O)NC(CC2CC2)C(=O)OC(C)(C)C)cc(F)c1 c1(C(=O)NCCC(CNC(C(C)SCCCC)=O)O)ccc2cccnn12 c1(C(N(C(CNC(COC)=O)C)C)=O)ccccc1OCc1cccc(Cl)c1 C(CCC(N)=O)(C(=O)NC(C)(C)CCNC(c1cnnc(O)c1)=O)N(C)C Cc1ccc(C(=O)NC(c2ccccc2)C(C)NC(C2C(C)(C)C2(C)C)=O)nn1 C1(C(=O)NCC(C)(C(C)C)NC(C2C(OC(C)=O)C2)=O)CC2(C1)CC21CC1 C#Cc1cccc(C(C(=O)NCC2CCOC2)NC(C)C2=CCN(C)CC2)c1F CC(CCCCNC(=O)CC1CC=CC1)NC(=O)C(C)(F)F C1(NC(C(C)C)=O)CC2CN(C(C3CCN(Cc4ccc(F)cc4)C3)=O)CC2C1 c1(C(=O)NCC2CC(O)(CNC(CNC(=O)NC)=O)C2)ccc(C#N)cc1O c1(C(=O)NCC(n2cc(-c3ccn(CCF)n3)nn2)C)c2c(nn1C)CCSC2 C1(CC)CCN(C(=O)C(c2ccccc2)C)C1C(=O)N(CC(=O)OC)CC c1(C(=O)NC2CCC3CN(C(C4(F)CCC4)=O)CC3C2)ccc2nc(O)[nH]c2c1 S(=O)(=O)(c1ccccc1C1(C#N)CCC1)Nc1c(OC)cc(C)cc1 C1(NC(Cc2cc(C)sc2)=O)CCC(C)N(CC(=O)NCc2ccco2)C1 c1(CC(=O)NCC2(O)CN(C(=O)C=Cc3ccncn3)C2)cccnc1O C(=O)(C(C)(C)CNC(N)=O)NC1C(=O)C1CCNC(COC)C(C)C c1(C(=O)NCC(CNC(=O)C(=O)NCC2CC2)OC)c(Cl)n[nH]c1C C1(c2nn[nH]n2)(NCC=CC(=O)NCCC23CC(CO2)C3)CCCC1 N#CC(C(N)=O)NC(C1CC(NC(C2CCOCC2)=O)C1)=O N1(C(CCc2cc(C)no2)=O)CCC(NC(=O)CC2CC=CC2)C(F)C1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CCC(C(C)NC(c2ncncc2Cl)=O)CC1 C1(C(N(C2CCC(NC(C3C(C)OC(C)C3)=O)CC2)C)=O)CC(=O)NC(=O)C1 N1(C(c2cccc(C)c2)=O)CCN(C(c2csc(CO)n2)=O)CC(C)(F)C1 CCCCCCN(CCN(C)CC#N)CC.C1(c2ccoc2)C(=O)N1 c1(C(=O)NCC2(CNC(C(CC)OC)=O)CC23CCC3)cccc2[nH]cc(Cl)c12 C=CC(C)(C)CC(=O)NCCC(C)NC(=O)Cc1ccccc1CC(N)=O c1(C(=O)NC2C(NC(c3cc(O)cs3)=O)CCCC2)cc2n(n1)CCOC2 c1(C(=O)NC(CNC(CCC(C)OCC)=O)(C)C(C)C)cc(O)ccc1F CC1(C)CCOC(CC(N2CCC(F)(CNC(c3ccc(F)cc3Cl)=O)C2)=O)C1 C1(C(=O)NC2C(CNC(CC(C)n3cccn3)=O)CCCC2)C(F)(F)C12CCC2 c1(C(=O)NC2CC(C)(C)CN(C(=O)CN=S(C)(C)=O)C2)cc2nc(F)ccc2o1 N1(C(=O)NC(c2ccc(C#N)cc2)C(C)C)CC2(CC2)c2ccc(Br)cc21 N1(C(C(C=C=C)C)=O)CC(NC(c2ccn3nccc3c2)=O)CC2(CC2)C1 C1(NC(COC(C)C)=O)CC2CN(C(=O)CCc3ccccc3F)CC2C1 C1(O)(CCNC(C2CC3CCC3C2)=O)CCN(C(C2COCOC2)=O)CC1 S(=O)(=O)(c1ccc(Cl)cc1)N1C(NC(c2ccccc2[N+](=O)[O-])=O)CCCC1 N1(C(c2n(C(C)C)ncc2Cl)=O)CCN(C(C2(O)CCC2)=O)C2(CCC2)C1 C1(CC(C)NC(=O)C(C)n2ccnc2)CCN(C(=O)CCOC2COC2)CC1 C(=O)(C(CNC(=O)CC1CCOC1(C)C)C(C)(C)C)NCC(CC)F c1(C(=O)NCCC2(OC)CN(C(=O)Cc3cnn(C)c3)C2)c(C)cnn1C c1(CC(=O)NC2CCCN(C(C=C(C)Cl)=O)C2C)coc2ccc(F)cc12 c1(CCC(=O)NCCCCC2(NC(=O)NC3C(C)C3)CC2)nccn1C n1(CC)nc(C(=O)NC2CN(C(C3CC3CNC(C)=O)=O)CC2(C)C)ccc1=O C(=O)(C1CCCc2n[nH]cc21)NC1C2CN(C(C=Cc3c(C)ncs3)=O)CC1C2 N1(C(CC2CCC(C)CC2)=O)CCC(NC(c2cc(C#N)c[nH]2)=O)C12CCCC2 C1(O)(C(C(=O)OC)(C)C)CCN(S(=O)(=O)N2CC(O)Cc3ccccc3C2)CC1 N1(Cc2scc(CCN(C(C)=O)CCN)c2)CCOCC1C(C)(C)C C1(=CC(=O)NC(C(C)C)C(C)NC(C2CCC(C)(C)OC2)=O)CN2CCC1CC2 C(=O)(C(CC(F)F)N(C)C(c1cc(CC2CCCCC2)[nH]n1)=O)N1C(CC)CC1 C1(C(=O)NC2CCN(C(=O)CCC3CC3)CC2)CC2C=CCC(C1)C2 C(C)(C(C)(C)CO)n1cc(C(C(=O)Nc2nc(C3CCC(C)C3)on2)(F)F)nn1 CN1CCC2(CN(c3ccnc(NCC(N4CCOCC4)(C)C)n3)C2)C1 C1(C)(CNC(C(C)N(C(C)=O)C)=O)CCN(C(c2c(C(F)(F)F)cnn2C)=O)C1 CCC(CCC(=O)N1CCC(CN(C(=O)Cc2cnn(C)c2C)CC)C1)OC c1(OC)ccc(Cl)c(C(N2CCCC(N3CCCC3(C)C)C2)=O)c1F C1(c2ccc(F)cc2)(NC(=O)NCCCc2cccs2)CCCCC1 c1(COCCNC(=O)CC2(C(C)=O)CCOC2)ccccc1CNC(N)=O.C1CO1 C1(NC(=O)COC2CCCC2)COC2(CCN(C(c3cc(F)cs3)=O)C2)C1 C12CCN(C1=O)n1cc(nn1)C2SCc1nc(COC)on1.c1(C2CC2)nc[nH]n1 C=C1CCC(C(=O)NC(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)CC1 c1(C(N2CCC(OCCNC(c3cnc(C)s3)=O)C2)=O)c(F)cc(Cl)cc1F N1(C(C)=O)CCC2(CCCN2C(=O)C(CC(F)F)C2CCCC2)C1 C1(C)(CNC(c2ncc(CC)cn2)=O)CCN(C(c2ccc(C3CC3)s2)=O)CC1 c1(CC)cccc(NC(C2CN(C(=O)CC3C=CCC3)CC2C(C)C)=O)c1 n1(CC(=O)NC2CCC(CNc3cc(O)nc(O)n3)C2)nnc2c1CCCC2 C1(NC(Cn2ncc(C)c2)=O)COCCN(C(C2(CF)CCC2)=O)C1 Cc1c(C(N2CCCC(F)(CNC(C3(O)CCC3)=O)C2)=O)oc2c1C(=O)CCC2 c1(C(=O)NC2C(NC(Cc3cc(C)sc3C)=O)C2)c[nH]c2ncccc12 N1(C(c2csc(C(F)F)n2)=O)CC2CCCC(C1)N(C(=O)C=CC=C(Cl)Cl)C2 N1(CC(C)C)N=C(C(=O)NC2(CO)CCCN(C(=O)CC(C)SC)C2)CCC1=O C1(CNC(=O)CCc2ccc(Cl)s2)CN(C(C2CCC(F)(F)C2)=O)CC12CC2 C(=O)(C(F)C(F)(F)F)N(CC(C)O)CCNC(c1c[nH]c(-c2ccccc2)c1)=O c1(CN2CCC(C(C(=O)NC(c3onc(C)n3)C)C)CC2)ccc(C)cc1Br C#CCC(C(=O)NCCC(O)COC)NC(c1nnc(S)n1C)=O c1(C(c2n(CCCCCC)nnn2)NC2CC2C2CC2)ncc(C)cc1Cl c1(CN)ccccc1SCCC(=O)NCc1ccc(Cl)s1 C(=O)(C(C)(C)S(C)(=O)=O)NCCC1N(C(c2[nH]cc(OC)c(=O)c2)=O)CCSC1 CC1Oc2ccccc2OC1C(=O)NCC1CCCN1C(=O)C1=C(Cl)CC1 Cc1c(C(=O)NC2CCN(C(c3ncc(Cl)cc3F)=O)CC2)[nH]ccc1=O C1(NC(c2c(C)nc(C)o2)=O)CN(C(C2COCC2(C)C)=O)C2(CCC2)C1 N1(C(C(CC(C)C)C)=O)CCC2CCC(C1)N2C(c1ccc2c(n1)NCC2)=O CC(C)(C(=O)NC1C2CN(C(C3CCN(CCO)C(=O)C3)=O)CC12)C(F)F c1(OC)cc(C)c2c(c1)C(NC(c1cccc(N=S(C)(C)=O)c1)=O)C(=O)N2C N1(C(c2c(O)c(F)cc(C)c2N)=O)CC2(CCCN(C(=O)CN(C)C)C2)C1 N1(C(C(CSC)OC)=O)CC2CCCC(C1)N2C(c1ncnc2c1OCCO2)=O CCC(C)C(O)C(C)C(=O)N(C(C)C(=O)Nc1cccc(CO)c1)C1CC1 C1(CNC(C2CC(C)(C)OCC2)=O)C2CCCC1N(C(=O)C1=NNC(=O)C1)C2 c1(C(C)(C)NC(C(=O)N(C(COC)Cc2ccccc2)C)=O)cccnc1 c1(C(N(c2c(N)cc(Cl)nc2)c2cc(Cl)cc(Cl)c2)=O)ccc2nnnn2c1 Cn1[nH]c(C(F)F)nc1=NC(=O)C(Cc1ccc(C(F)F)cc1)CN c1(C(N2C(CNC(c3c(C)nc[nH]3)=O)C3CCC2C3)=O)noc2c1CCCC2 N12CC3(CCN(CC3)C(=O)C3(CC3)C1=O)C2.c1(C(C)(C)C)ccnc(F)c1F C1(C(=O)NC2C(CNC(C(CC)N3CCCC3=O)=O)C2)CN(C)CC1C(F)(F)F c1(C(=O)NCC2(C)OCCN(C(C(C)OCC3CC3)=O)C2)cnn2ccccc12 N1(C(C(C)=CC)=O)CC=CC(NC(c2cnc(NC)cn2)=O)C1 CC(C)CC(C(=O)Nc1cnn(C(C)C)c1)NC(=O)C(C)O N1(C(C2C(=C)C2)=O)CCN(C(c2cnc(Cl)c(N)c2)=O)C(CC(F)F)C1 C1(NC(CC(CC)SC)=O)CN(C(c2cccc(C#N)c2)=O)C2CCCC12 N1(C(c2cnn(C3CCOCC3)c2)=O)CC2(CCCC2NC(C2(CF)CC2)=O)C1 N1(C(C(=O)N(C(C)C)C)C)CC(C)(C)CCC1CNC(c1cnn2ccsc12)=O c1(C(=O)OC)cc(N2CC(CCCCNC(c3conc3C(C)C)=O)C2)ncn1 c1(-c2ccc(N(C)C)cc2F)ccc(S(=O)(=O)N2CCC(O)(COC)C2)c(Cl)c1 N1(C(C2(C)N(C(c3c(C)n(C)nc3)=O)CC=C2)=O)CCOC2(CCC2)C1 c1(CNC(CCOC2CCN(C)CC2)=O)nn(C)c2c1CN(C(=O)C(F)F)CC2 CC(C(=O)NCC1CCN(C(=O)CCNC(=O)OC(C)(C)C)C1)C(F)(F)C(F)F CC(C)(O)C#CC(=O)N1CCC(CCC(=O)N(CCCO)C2CC2)C1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CN(C(c2cn(CCC)nn2)=O)CC(O)C1 c1(NC(C2(C)CC2)=O)c(-c2cnn(CS(C)(=O)=O)c2)ccc2c1OCO2 c1(CNC(C2(C(F)(F)F)CC(C)(C(=O)OC)C2)=O)cnc(C(F)F)cn1 N1(C(CC2(C)CCCCC2)=O)CCOCCC1C(=O)NCC1CCN(C2CC2)C1 C12CCCN(C1)C(C)C(=O)N2.C1(C(=O)OCC)CCOC1C(F)(F)F CCCCC(CNC(=O)C=Cc1cccs1)NC(=O)Cn1ccc(C(F)F)n1 c1(C(=O)NCC2CC2CNC(c2cnnn2C2CC2)=O)ccc(-n2ccnn2)cc1 N1(C(C2C(c3ccc(C)s3)C2)=O)CCN(C(=O)Cc2cnccc2C)CC(O)C1 C#Cc1ccnc(C(=O)NC2CCCN(C(=O)CC(=O)NCC3CC3)CC2)c1 Cn1cccc1C=CC(=O)NC1COCCC1NC(c1cscn1)=O c1(CCNC(C(C)OCCn2ccnc2)=O)c(F)cccc1F N1(C(C)=O)CC(C)CN(C(c2cccc3nc(CC(C)C)[nH]c23)=O)C(C)C1 C12(NC(C3CCN(C(c4ccnc(O)c4)=O)CC3)=O)CCC(CC1O)C2 C1(C)(NC(c2c(C)[nH]cc2)=O)CCN(C(=O)C(Cc2ccsc2)NC=O)C1 N1(C(C2C(COC)C2)=O)CCCC(NC(C2CC=C(C)CC2)=O)C1 CC1(C)CC(CNC(=O)COCc2nccs2)CN1C(=O)C=C(Cl)Cl CCC(CC(=O)NCCC1CC(F)(F)CN1C(c1cc(N)ccc1C)=O)C(F)F C(=O)(C(O)CC(C)(C)C)NCCC1(NC(C2N(C(C)=O)CCC2)=O)CCC1 N1(C(c2cn(CC(CC)O)nn2)=O)CC=C(CCNC(C2SCCS2)=O)CC1 N1(C(C=CC)=O)CC2CCOC2(CNC(=O)Cc2cncnc2O)C1 CCC(C)(CNC(=O)CCCC(C)NC(C1CCC(=O)O1)=O)C(N)=O C12(NC(C3CCN(C(C)=O)C3)=O)CCC(CN(C(c3ccc(C)cc3Cl)=O)C1)C2 CCCCC(F)(F)C(=O)N1CC2(CCC2)CC1CNC(=O)CC1CC1 c1(C(N(CCC(=O)NCC#CCOC)CCO)=O)ccc(C#N)[nH]1 C(c1cnccc1C)=CC(=O)NC(CN(C(C(C1CCCC1)OC)=O)C)C CC(C)C(F)(CNC(C1CCCC(=O)CC1)=O)C(=O)NCCCCC(N)=O C1(C)(CC)CCNC(=O)CC(=O)N1.C=CCNC(C)=O CCC(C)C(C(=O)N(C(C)CCSC)C)NC(=O)C=CCOC CS(=O)c1ccc(CC(=O)NC2(NC(=O)C(C)(O)C(C)(C)C)CC2)cc1 c1(CN2CCC(NCc3c(C(=O)O)nco3)CC2)cc(Cl)cc(Cl)c1 N1(C(C(CCC2CC2)NC(C(C)c2cc[nH]n2)=O)=O)CCOC2(CCC2)C1 C(CCC(C)CC(=O)NC12COC(CNC(c3cn[nH]c3)=O)(C1)C2)=C(C)C c1(SCCC)ccc(C(=O)NC2CC(N(C)C(c3cn(CC)nc3C)=O)C2)cc1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CC2CCC(CNC(c3cc[nH]n3)=O)C2C1 CC1(C)CC(NC(=O)CCCNS(C)(=O)=O)CN(C(c2ccc(=N)[nH]c2)=O)C1 C(C)(C(=O)NCC(=O)NCCN(CCC(F)F)C)OCC c1(C(=O)NC(C23CCC(CC2)C3)CNC(CCOCC)=O)cn2c(n1)COCC2 c1(C(N(CCNC(C2N(C)C(=O)OC2)=O)C2CC2)=O)ccccc1C#N Cc1nc(NCC(CO)C(F)(F)F)cc(NCc2nnc(C(C)(C)C)s2)n1 C(=O)(CC(C)C(F)(F)F)N(CCOCCC(=O)NCC(CC)(C)CC)C c1(CC=C)cn(CCCC(=O)NCc2ncn(CCCCC)n2)nn1 N1(C(c2cc(C)cc(O)c2)=O)CC2CCC(NC(=O)C=C3CCN(C)C3)CC2C1 CC1(C)C2CCC1(C)C2C(=O)NCCCCNC(c1cc(C2CC2)[nH]n1)=O c1(C(=O)NC2C(NC(C=C(C)c3ccco3)=O)CCC2)cc(C)cc(Cl)c1 c1(NC(C2N(Cc3nc(C)[nH]n3)CC(O)C2)=O)cccc(Cl)c1F C(=O)(C(CC=C)CC(C)C)NC(CC=C)CNC(c1cc2c(C)nn(C)c2s1)=O CC1CC(NC(c2cc(Cl)c(Br)[nH]2)=O)CN1C(=O)CCc1ccoc1 c1(C(=O)NC2CCN(C(Cc3cccc(CC)c3)=O)C2)cc2oc(Br)cc2[nH]1 c1(C(=O)NCC2N(C(CC(C(C)C)C)=O)CCCC2)ccc(C#N)c(F)c1 C1(NC(C(C)(C)OC(C)=O)=O)CCCCC1NC(=O)C(F)CC1CCC1 c1(C(N2CC(OC)CC(NC(C(CC)COC)=O)C2)=O)ccc2oc(O)nc2c1 CCC(CC)CCC(=O)NCC1CN(C(=O)CC(=O)NCC)CCO1 C(=O)(CS(=O)(=O)C1CC1)NCCC1(CNC(Cc2c(Cl)cn(C)n2)=O)CC1 C12(NC(=O)NC)CCCC1CCN2C(c1n[nH]c(C)c1Cl)=O.C12CN(C1)C2=O N1(C(C2(NC(C)C)CC2)=O)CC(n2cc(-c3ccc(C(C)O)cc3)nn2)C(C)C1 C(C)(C(=O)N1CCCCO1)(N(C(CCc1cc(C)[nH]n1)=O)C)C1CC1 C1(CNC(COCC(C)C)=O)CC(CNC2(c3nc[nH]n3)CCC2)C12CCC2 c1(C(=O)NC2CCC(NC(C=C(C)C3CC3)=O)C2)cc2c(Cl)cc(Cl)cc2[nH]1 C(CCC(O)C(=O)N1CC(CO)C1)NC(c1c(OC)nccn1)=O CC1(C(=O)NCC2(CNC(c3ccoc3)=O)CC2)CCn2ccnc21 C1(C2CCCN(C(C3CC(C)(C)O3)=O)C2)(NC(c2c(C)ccnn2)=O)CC1 C(=O)(C(C)C1OCCc2ccccc21)N1CCC(COC)(CSc2ccccc2)C1 N1(C(c2n(CCOC)ncc2)=O)CC(COCC(O)COC)OC(=O)C1 C1(NC(CCCSC)=O)CC2CC(NC(=O)C(C)OCC3CC3)CC12 C1(NC(C(CCC)=CC)=O)CN(C(=O)C(C(C)C)NC(N)=O)CC12CCOCC2 C1(F)(CNC(C2CN(C(C)C)C2)=O)CCN(C(=O)CC2CCC(=O)NC2)C1 c1(NC(C2N(C(c3c(CC)nc(C)o3)=O)C(C3CC3)CC2)=O)ccc(F)nc1C C(CC(C)(C)C(=O)N(C)Cc1ncco1)NC(CCC)=O C=CCC(C(=O)N1CCC1(C)CC(=O)NC(C(=O)OC)CO)OC Cc1cc(=NCCn2cc(Cl)cn2)[nH]c(N(C)Cc2nc3ccccc3n2C)n1 N1(C(c2c(C)nc(O)[nH]2)=O)CC(CCNC(c2c(Cl)cccc2Cl)=O)OC(C)C1 C1(C(=O)NC2CCN(C(C(c3ccc(C)cn3)(F)F)=O)C2C)COCC(C)(C)O1 Cc1cnc(CCC(=O)N2CC(=C(F)CNC(=O)CN3CSCC3=O)C2)[nH]1 N1(C(=O)COCC2CC2)CCC(=CC(N2CC3CC3C2)=O)CC1 c1(NC(C2C(C(=O)NCC(C)(C)C)C2)=O)cc(Cl)c(Br)c(Cl)c1 N1(C(C(CC=C)CNC(c2cccn(C)c2=O)=O)=O)CC(=O)NC(=O)C1C N1(C(C=C(C)C(F)F)=O)CCC(CC(=O)NCc2nc(C)co2)C1 c1(NC(=O)NCc2cc(Oc3ccccc3)ccn2)coc2c1C(O)CCC2 C(=O)(C#CC1CCOC1)N1C(C(=O)NC2C(C#C)CCC2)CCCC1 c1(C(=O)NC(C(C)NC(c2c(CC)noc2)=O)C)cccc2nc(O)n(C)c12 c1(C(=O)NC(C2CCN(C(C3CC(OC)C3)=O)C2)C)cncc2ccsc12 CCC1=C(C(=O)NC2CC(C(=O)NCCSc3ccccc3)C2)CCCO1 Cc1cc(CN2CC3CC3(C(=O)N=c3nc[nH]s3)C2)cnc1Cl C1(NC(c2cccn(C(C)(C)C)c2=O)=O)CC2CC1CN2C(=O)C=CC1CC1 Cc1ccc(CCC(=O)NC(C)CN(C(=O)CCCC(C)O)C)c(C)c1 CCCCC(CC(=O)N1CCC(O)C(O)C1)NC(=O)CCC(F)(F)C(O)C C(C)(C(=O)N=c1ccn(C)[nH]1)NN(S(c1cccc(OC)c1O)(=O)=O)C CC(C)(CC(F)F)C(=O)NC1CCC(C)(CNC(C2C=CCS2)=O)C1 Cc1cc(=NC(=O)CC2CCCN(C(C3CC(C(C)C)=NO3)=O)C2)[nH]n1C N1(C(C(CC)CC)=O)CCCN(C(c2cc3n(n2)CCCO3)=O)CC1C CC1(C)CC(C(=O)O)(NC(=O)Cc2cnsc2)CO1 C1(F)(CNC(COC(=O)C2CC2)=O)CCCN(C(=O)CCOCC(F)(F)F)C1 CC1C=C(C(=O)N(C)CCC2CCN(C(c3cncc(F)c3)=O)CC2)CC1 N1(CC)CC(CNC(=O)CN(C(=O)C(c2ccc(F)cc2)F)C2CC2)OC1=O C(C(C)(CC)C(=O)N=c1ccn(C(C)CC)[nH]1)NC(CCCC#C)=O c1(OCC)ccc(C(=O)NCC2CCCN(C(c3cnc(C)n3C)=O)C2)cc1 c1(C(C(=O)Nc2cnn(C)c2CC)N(C2CCCCC2)CC)ccc(O)c(OC)c1 N1(C(c2cc(CC)on2)=O)CC2COCCC2(NC(=O)CC2CCCCC2)C1 C(=O)(C1=CCC(F)(F)CC1)NCC(C)(CO)NC(c1c(OC)ccc(O)c1)=O C1(CNC(C2C(CCOC)C2)=O)CCCCN(C(=O)Cc2nccn2C)CC1 Cc1ccc(C(F)(F)C(=O)NC2(CCNC(C3(C(F)F)CCC3)=O)CC2)cc1 CC1(C)CC1(C)C(=O)NCCc1cc(C(=O)NCCN2CC(CF)C2)no1 Cc1ccc2cc(C(N3CCN(C(=O)C4=C(Cl)CCC4)CC(C)C3)=O)ccc2c1 CC(C)CC(C)(O)C(=O)NCc1nc(C(=O)NC2(C)CCSC2)co1 C1(C(=O)NCC2(F)CC(NC(=O)C=CCO)C2)Cc2c[nH]cc2S1(=O)=O c1(C(=O)NCC2(C)CCCN(C(C3CC(F)(F)C3)=O)C2)ncnc2c1CCCC2 Cc1cc(CC(=O)NOCC(N2CC(O)(C#CBr)C2)=O)cc(F)c1 CC(C)CCCCN(C1COCC1n1ccnc1)CCN1CCN(C)CC1 C(=O)(C(CNC(=O)CC(C)(C)C#N)CC(C)C)NC(CC)CCO N=c1nc(CC(N2CCC(C(=O)Nc3cnn(CC(N)=O)c3)C2)=O)[nH][nH]1 Cc1cccc(OCC(=O)NC(CNC(c2ccc(Cl)cc2F)=O)C2CC2)c1C CC1(C)COCCC1C(N1CCC(CNC(C2CCC3CC2CO3)=O)(CF)C1)=O c1(NC2(CNC(c3cnc(SC)nc3O)=O)CCCC2)ncnc2c1ncn2C Cc1cc(C(=O)NC2CCCCC2CC(=O)N(CC(C)(C)O)C)ccc1F C1(O)(CNC(C2CCC(CC)CC2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1 C1(C(=O)NC2CN(C(C3(C)CC(=C(F)F)C3)=O)CC2C(F)F)Cc2nccn2C1 Cc1ccc2snc(NC(C)C(C)CCCCl)c2c1 N1(C(Cc2ccc(SC)cc2)=O)CCOC2(CCS(=O)(=O)C2)C1 Cn1nnc2c1CCC(C(=O)NCCCCCNC(=O)CC1COCC1O)C2 n1(CCCC)nnnc1C(CCC1(C)CC1)N(C1(CCC(F)(F)F)CC1)CC C1(C(=O)NC2CC(CNC(C3CC(CCC)C3)=O)C2)C(Cl)(Cl)C12CC2 N1(CC(CC)NCc2ncnn2Cc2cccc(Cl)c2)CCCC(N(C)C)C1 CC1CN(C(c2cn3ccccc3n2)=O)CC(C)N1C(=O)CN1CSCC1=O N1(C(c2cn(CC=C)nc2)=O)CC2CC1CN(C(=O)CCS(N)(=O)=O)C2 c1(C(=O)NCC2(C)C(NC(CSC)=O)CCC2)cc2cccc(Cl)c2s1 c1(C(N(C2CCCCC2NC(C2CC=CC2)=O)C)=O)c(F)cc(Br)cc1F C1(CNC(c2cnn(C3CCOCC3)c2)=O)CCC(NC(C2CS(=O)(=O)C2)=O)C1 C(c1ccc([N+](=O)[O-])s1)=CC(N1CC(CNC(CSCC)=O)C(O)C1)=O c1(C(=O)NC(C)CNC(=O)C(F)(F)C(F)F)cc2ccc(Cl)cc2[nH]1 C(=O)(C(C)(C)C(C)(C)O)NCCC1(NC(C(c2cc(F)cc(F)c2)C)=O)CCC1 CC1C(C)N(C(c2c(Cl)sc3nnsc23)=O)CCN1C(c1cncn1C)=O c1(C(=O)NCC2CCCN(C(c3c(CC)con3)=O)CC2)c(Cl)ccc(F)c1C S(=O)(=O)(c1ccc(C(=O)NCC(C2CCC2)NC(=O)COCCCF)cc1)N(C)C CCC(C)(C)C(=O)C(=O)NCC1CN(C(C2CCCN2C=O)=O)CC1(F)CO CC(C)C(C)C(C(=O)O)NC(c1cc(=O)c(Br)c[nH]1)=O Cc1c(O)ccc(NCC(O)CN2CC(C)OC(C)C2)c1C C(CC1=CCN(C(C2CCc3nn[nH]c3C2)=O)CC1)NC(C)=O CCCCC(C(=O)NCC1CCC1CO)NC(=O)CC(C)(C)COC O=C(CS(=O)(=O)c1ccccc1F)N1CCCC1CC1(Cc2ccc(F)nc2)N=N1 C1(NS(CC)(=O)=O)CCN(C(=O)C(C(C)C)NC2CC2(C)C)CC1C n1(OCc2n(CCS(C(C)C)(=O)=O)nc(C(C)O)n2)c(CO)nc2ccccc12 C1(CNC(CCC=C)=O)CN(C(c2ncccc2O)=O)C2CC12 C1(CC=C)(NC(C2CCCCC2)=O)CCCN(C(c2nccs2)=O)C1 CS(=O)(=O)C(C(=O)NCC1(CNC(=O)CN2CCCCC2)CC12CCC2)C1CC1 N1(CCC(=O)NCC2CCC(NC(CSC)=O)C2)C(=O)NC(C)(C)C1=O N1(CC)CC(C)N(C(=O)C(N2CCC3(CC2)OCCO3)=O)CC1(C)C n1(C(C)C)ncc(C(=O)NC(C2(O)CN(C(C3NC(=O)OC3C)=O)C2)C)n1 Cc1cnc(C(=O)NC2CCCN(C(=O)CC3(O)CCCCCC3)C2)cc1C C(=O)(C(C(=O)NC(C)CC(C)NC(=O)CCc1cc(C)on1)C(C)(C)C)OCC Cc1cc(Br)cc(C)c1CNC1(n2cc(CCCC(C)O)nn2)CCN(C)C1 n1(SC)ccc2ccc(C(c3nnnn3C)NC3(c4c(C)noc4C)CC3)cc12 C1(CC(=O)OCC(C2CCC23CC3)=O)CC2C=CC1C2 C(=O)(C1=NOC(C)(C)C1)N1CCC(CC(N)=O)(NC(c2n(CC)nnc2)=O)CC1 c1(CCNC(COCCC)=O)ccc(CNC(c2ccc(C)[nH]2)=O)cc1 c1(C(=O)NCC(CNC(c2c(OCC)ccs2)=O)F)cnc2c[nH]nc2c1 Cc1cc(S(=O)(=O)NC(C2CCOC(c3cccs3)C2)=O)c(C)c(S(C)(=O)=O)c1 C1(C(C(=O)NCC2CC2NC(=O)C=C2CCCC2)OCCOC)CC(F)(F)C1 C(=O)(C(CO)C(C)(C)C)NCC(CC(=O)N(C(C)C(=O)OC)CC)C C(=O)(C(C(C)(C)C)NC(N)=O)N1CC(F)(CNC(C=C(CC)CC)=O)C1 C1(O)(C(C(=O)NCC(CC)NC(C=C(CC)CC)=O)F)CCCC1 C1(C(=O)OCC)CCN(C(=O)CCCc2ccccn2)C(C)(C)C1 N1(C(c2c(C)cc(=N)[nH]c2)=O)CCC2(CCC2CNC(=O)C(O)C(F)(F)F)CC1 C=CC(C)(CCOC)C(=O)NCCCN1CCN(C(=O)C=CC2CCCO2)CC1 N1(C(c2ccc(C)c(F)c2)=O)CCCC2C1CCCCN2C(=O)C(O)CC(C)C C1(C(=O)OCC)CCCC(C(=O)N(CCCN(C(C2CC2[N+](=O)[O-])=O)CC)C)C1 Cc1ccc(F)c(C(=O)NCC23CC(NC(=O)C(CCO)N(C)C)(C2)C3)c1F C1(CNC(CC(=C)C)=O)CC2(CCN(C(=O)CCc3cnn(C)n3)C2)CO1 CC(c1cccs1)=CC(=O)NCCCC(C)NC(=O)C(C)(C)C1CCOCC1 Cc1cccc(C)c1NC(=O)C(c1cn[nH]c1)N(CCC(C)C)C1CC1 c1(C(=O)NCC2N(C(C(CC)O)=O)CCC2)cc(C)nc2c1cnn2CC N1(C(C(COCC)C)=O)CCC2(CNC(=O)Cn3ncn(C)c3=O)CCCC12 N1(C(CCCSC)=O)CC2C(NC(=O)C(c3ccc(C)s3)C)C2C1 CC1COC2(CCC2)CN1C(C1CC2(CCC2)CN1C(=O)C(C)C(F)F)=O Cc1cccc(C)c1CN(C(=O)C(=O)NC(C)C(C)S(C)(=O)=O)C CCC(C)(C)C(C)CC(=O)NC12CC(NC(=O)CSC3CC3)(C1)C2 C(CCN=C(NCCc1occc1C)N1CCN(C(C)C)C(=O)C1)OC(=O)NC c1(C(=O)NCC2CC(OC)CN2C(=O)C=C2CCC2)ccc2c(c1)CCOC2 CSC1=C(C(=O)N(C2CCN(C(c3cnnn3C)=O)CC2C)C)CCCC1 C=C(C)CN=C(NCc1cccc2c1OCC2)NC1CCS(=O)(=O)C1 c1(OC)ccc(O)c(C(N2CC(C3(NC(=O)CNS(N)(=O)=O)CC3)OC(C)C2)=O)c1 C(=O)(C(CCC)CC(C)C)N(C(CCC=C(C)C)C)CC.C1(CC(=O)N)CCOC1(C)C C1(NC(C(C)Cc2ccnn2C)=O)CCN(C(=O)CC2(O)CC2)CC1(C)C N1(C(CCCCCN(C)C(C2(C)CCCO2)=O)=O)CC2CCC(C1)N2C C1(C(=O)NCC2CCOC2)(OC)CCN(C(c2csc(Cl)n2)C2CC2)CC1 c1(C(=O)NC23CC(CNC(CC4N(C)C(=O)CC4)=O)(C2)C3)cnc2ccoc2c1 C1(N(CCOC)C(C2CS(=O)(=O)C2)=O)CCN(C(=O)C(C)C(C)C)CC1 c1(N(c2ncnc3ccsc23)C)nc(=NC2CC2C(N)=O)[nH]c2c1SCC2 c1(C(N(C)CCN(C)C(C2CCO2)=O)=O)ccc2nc(C(F)(F)F)[nH]c2c1 C1(C(=O)NCc2cc(C)sc2C)(COC)C=CCN1C(=O)C(n1cc(C)cn1)C C=C(Br)CC(=O)NCC1CCCN1C(c1ccnn1CC(C)C)=O Cc1ccc(Br)c(C(C)NC(C2CCOC2C#N)c2nnnn2CC2CC2)c1F N(C(=NCc1c[nH]c2cccc(F)c12)N1CCN(CC(C)C)CC1)C(CC)C c1(NC(CCNC(c2c(CC)onc2C)=O)C)ncnn2c(Br)ccc12 N1(C(=O)Nc2c(C=O)cccc2F)CCc2cnccc2C1 c1(NC(CC)=O)ccncc1C(=O)N(C)CC1CCN(CCN2CCOCC2)C1 N1(C(c2ccc(CC)cn2)=O)Cc2ccccc2CC1CNC(=O)C(Br)=C(C)C C1(NC(C2CCC(NC(COCCC)=O)C2)=O)CC2CC1CC21CC1 C(CCC(C)C(=O)NC1CC(C)N(C(c2cccc(CN=[N+]=[N-])c2)=O)C1)OC Cn1nc(CC(=O)NC2CCC(CCNC(=O)C(=O)NCC(F)F)C2)cc1Cl c1(CC)sc(C(N2CC(OC)CC2CCNC(=O)CC(C)(F)F)=O)cc1C N1(C(COCCC#C)=O)CCN(C(C2CC(C)OC(C)C2)=O)CC1C(F)F N1(C(C(=O)N(CC)Cc2noc(C(F)(F)F)n2)=O)CCCC(C#N)C1 C1(NC(C2CCCCC23CC3)=O)COC2(CCN(C(c3coc(Cl)n3)=O)CC2)C1 c1(C(=O)NCC(C2CC2)NC(C(COC)N(C)C)=O)cnn2c1NCCC2 C(=O)(C(CS(C)(=O)=O)c1ccccc1)Oc1c(C)cccc1.c12ccccc1o[nH]2 c1(C(=O)OCC)cccc(NCC)c1C.N12CC3C(C3C1)C2=O.N(CCO)(C(C)=O)CC#N N1(C(c2c(N)cn(C)n2)=O)CC(CNC(c2nncn2C2CC2)=O)C(F)(F)C1 C1(C(=O)N(CC(O)CF)C)(CC)CCCN1C(c1ccncc1Cl)=O C1(NC(C(C)(C)NS(C)(=O)=O)=O)COCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 c1(C(=O)OCC)cccc(C(=O)N(CC(C)NC(C2CCC2(C)C)=O)C)n1 N1(c2snc(C)n2)CC2CC(NC(c3ccncc3Cl)=O)CC2C1 C1(C2CCN(C(=O)CCCC(N)=O)CC2)(NC(CC(C=C)c2ccccc2)=O)CC1 C(CN=c1nc2c(cnn2C)c(NCC2CC(C)(C)CO2)[nH]1)OCCN(C)C N1(C(C(C)NC(=O)NC)=O)CC2CCC1C2NC(=O)Cc1nn(C)cc1Cl N1(C(CCC)=O)CC(OC)C(N2CCN(C(c3ccncc3N)=O)CC2)C1 Nc1c(C(N2CCCC2C2CCN(C(C3CCCCC3)=O)C2)=O)ccnc1Br c1(C(=O)NC2C(CNC(CCC(=O)OC)=O)CC2)cc2c[nH]nc2cc1C CCC(C)(O)C(=O)N1CCC(CNC(=O)CN2CCC(O)CC2)CC1 c1(C(N2CCN(C(c3n(CC)nnc3C)=O)CC2)=O)ccc(C2CC2)nc1C c1(SCC)ccc(C(N2CCC(NC(C3CCCN(CC)C3)=O)C2)=O)cn1 N1(C(c2c(C)cc(N)cn2)=O)CCOC2CN(C(c3cccn(C)c3=O)=O)CC12 C1(NC(=O)Nc2c(CSC)c(C)nn2C)CCc2nc(=N)[nH]cc2C1 c1(C(=O)NC2CC(NC(c3nc(C(C)OC)oc3)=O)C2)n[nH]c(C)c1O CC1CN(C(=O)CC23COC(C)(C2)C3)CCC1CNC(C1CN(C)C1)=O C12(CNC(c3ncn(CC)c3)=O)CCC(NC(C3CCCC(O)C3)=O)(CC1)CO2 C1(c2cccnc2)(C(=O)NCC(F)(F)F)CCCC1.O=C1CNCCCN1 C1(C(C)C)CN(C(c2ncnn2C(C)C)=O)CCN1C(C1C(C2CC2)C1(F)F)=O c1(C(=O)NCC2C(C)CN(C(C3CC3(C)C)=O)C2)cc2n(n1)CCC2 N1(C(c2c(CSC)cccn2)=O)CCC(C)CC1CNC(=O)Cn1ccnn1 N1(C(CCC(=C)Br)=O)CC(NC(=O)CCc2cnn(C)n2)CC12CCC2 c12cn(nn1)C(C)CNC(=O)C21CCC1.c1(C(C(=O)O)OC)ccccc1 c1(C(=O)NC(C)CNC(=O)CCCSc2nnnn2C)cc(CSC)nn1C CC1(C)CC(CNC(=O)CC2CCC3CC23)N(C(C2CCN(CCO)C(=O)C2)=O)C1 N1(c2nccc(NCCCn3c(C)ncc3)n2)CCc2cccc(CO)c2C1 C1(Sc2cccc(-c3c(CCN4CC(C)OCC4)csc3)c2)CS(=O)(=O)C1(C)C C1(CNC(C2C(CNC(C3CC(C#C)(O)C3)=O)CC2)=O)CCC(=O)NC1C C1(C(=O)NC(c2nc(C)[nH]n2)C)CC(=O)CN1C(=O)CC(=O)OC(C)(C)C C1(C(=O)NCc2cn(CC)nc2)CC(=O)CN1C(C1CCN(C(C)C)C1)=O C1(NC(C(C)=C2CCC2)=O)CCN(C(=O)CN(C)CCO)C1C N#Cc1ccsc1C(=O)NCC1CCC1C(=O)NCCc1nccs1 C1(CNC(COCCCC)=O)CC2(CC2)CN1C(=O)C(c1ccc(F)c(C)c1)=O c1(CC(C)NC(N2CCN(C3CCN(C)C3=O)CC2)=O)ccc([N+](=O)[O-])cc1 c1(C(N2C3CN(C(=O)CSCCC(F)(F)F)C(CC3)C2)=O)cnn2c1CCCN2 C1(C(N2CCC(F)C2)=O)CCCN(C(=O)Cc2cc[nH]n2)C1 c1(NC)ccc(C(=O)NCCC(C)N(C)C(c2occc2C)=O)nc1 Cc1[nH]nc(Cl)c1C(N1CC(F)CC1CNC(=O)C(C)SC(F)(F)F)=O C1(NC(c2ccc(CN(C)C)o2)=O)CCOC12CCN(C(=O)C(C)(C)C)CC2 C=CCCC(CC(C)C)C(=O)NCC1(C)CCCN1c1ncc2ncnc-2[nH]1 c1(C(=O)NC2CCC(NC(=O)CCc3cnc(O)[nH]3)C2)ccccc1[N+](=O)[O-] N1(C(C(C)Sc2nncn2C)=O)CCN(C(=O)CC2OCCO2)CC1 C1(CC(=O)N(C(C)CCNC(=O)CNC(=O)C(C)(C)C)C)CC(C)(C)OC1=O C(=O)(C(C)C(C)C(C)(C)C)N1CCCCC(NC(Cc2cccc(C)c2Cl)=O)C1 Cc1ccc2sc(N(C)CC3CCCCN3C(C3(C)CCC(C)C3(C)C)=O)nc2c1 c1(NCC(CO)NC(c2ncc[nH]2)=O)cc(-n2ccnc2)ncn1 N1(CC(Cc2ccccc2)N(C)CC2CCOC2)CC2OC(=O)OC2C1 c1(CC(N2CC(O)(C(C)NC(c3cscn3)=O)C2)=O)cc(F)cc(Br)c1 C#CCC(C(=O)NC(C(=O)NCc1ccnc(CC)c1)c1ccco1)C1CC1 CON1CC(C(N2CCC3CC23C(=O)NCc2cccc(O)c2F)=O)CC1=O.C C(COc1ccccc1)(C(=O)N1CCC(CNC(c2nocc2F)=O)C1)OC c1(C(N2C(CNC(CC=CC=C)=O)CCC2)=O)cnn(CCC)c1Cl N1(C(CO)=O)CCC(COCC)C1.C1CO1.C(=O)(C1CC1)NCC Cc1[nH]c(C)c(C(=O)NC(c2ccc(F)cc2)CNC(=O)CCCN(C)C)c1C S(=O)(=O)(c1ccc(NCCCF)cc1Br)N1CC(CC)OC(C)C1 C1(CCC)CC(C(=O)OC(=O)C(C)(C)COCC)CCO1 c1(C(N(C(CNC(CN(C)CC)=O)C)CC)=O)nc2sc(C)cn2c1C C(N=c1[nH]nc(SC(F)(F)F)s1)c1cc(O)ncc1 C1(NC(C(C(CC)O)C)=O)CCCCC12CCCN(C(C1CC(=O)N1)=O)C2 O=C(C#Cc1ccccc1)N1CC2CCC(C1)N2Cc1c(I)ccnc1Cl CCCC(C(=O)NC(C(=O)NCCC1CC1)C(=O)OCCC1CC1)C(C)C S(=O)(=O)(c1cc(C(=O)O)ccc1F)N1CC(C(F)(F)F)CC(C(N)=O)C1 c1(C(=O)NC23CN(C(C4C(C)C4C)=O)C(C2)C3)ccc2ccccc2n1 C1(C(=O)NCC2CC(F)(CNC(CS(C)(=O)=O)=O)C2)OCC2COCCC12 C1(CC)(NC(C(=O)NCCNC)=O)CCCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 c1(C2CCN(C(c3nc(-c4ccc(F)nc4)no3)C)C2)ccnc(Cl)c1 C1(NC(=O)OC(C)(C)C)CC2(C1)CC2C(=O)N(C1CC2CCCC12)C1CC1 c1(C(=O)NCC2(F)CN(C(CC3CCCN(C)C3)=O)C2)n[nH]c2c1CCSC2 C(=O)(CCC(=O)NC(C1(O)CN(C(=O)CCc2cc[nH]n2)C1)C)NCCC c1(C(N2CCC(C(=O)NC)C2)C(=O)NCCOC)nc2cnccc2s1 C1(Nc2c(C)c(NC3CCCS(=O)(=O)C3)ncn2)CCn2c(C)cnc2C1 C=CC1(CC(N2CC(CNC(c3ccc(SC)o3)=O)(COC)C2)=O)CCCCC1 Cc1nc(F)ccc1CNCC1(C(=O)Nc2ncc(Br)cc2Cl)CC1 N1(CC(C)C)CC(C(=O)NC2CC(C)(NC(=O)Cc3ccc(Cl)cc3)C2)CC1=O CCCCCC(=O)NC1CC(CNC(=O)Cc2ccc(C)nc2)C1(C)C N1(C(=O)C2CC2)CCC2C(CCCN2C(=O)Cn2cccc2)C1 C1(N2CCC(N3CC(C)(C)C3)C2)CN(Cc2ccccc2)C(C)(C)C1 c1(C(=O)NC(C(C)NC(c2nc(CC)oc2C)=O)C)c(Cl)ccnc1C N1(C(C2CC(C)OC2)=O)CC2CC(NC(=O)C(CO)C(F)(F)F)CC(C2)C1 CN1CCOC(C(=O)NC2CCCC2CN(C)C(C2(CO)CCC2)=O)C1 c1(C(=O)NCC2C(C(=O)NC(C=C)CO)OCC2)cc(O)ccc1F C1(NC(C=C(COC)C)=O)CN(C(C2(Cc3ccc(O)cc3)CC2)=O)C2CC12 N1(C(=O)Nc2ccc(Cc3nccs3)cc2)C2CCC=CCC1CC2 C(c1ccc2c(c1)CCO2)=CC(=O)N(CCN(C)CC)CCOC c1(C(N2CCC(CCn3ccnn3)C2)C(=O)NC(C2CCCO2)=O)ccc(Cl)o1 c1(C(N(C)CC2CCN(C(C3CCC(C)(C)O3)=O)C2)=O)ccc2nc(O)[nH]c2n1 C1(C2CC2)(C(N2CCC(O)(CCNC(c3ccoc3Cl)=O)C2)=O)CC=CC1 Cn1cc(-c2cscc2C(N2Cc3cccc(F)c3C2)=O)c2ccccc12 N1(C(C(C)N(C)C)=O)CCC(NCCCC2CCCCC2)C(C)C1 c1(C(=O)NCCN(C(=O)C=Cc2ccsc2Br)CC)cnc(C)n1C c1(C(N(C2CCN(C(=O)C(=Cc3cccs3)C)C2)CC)=O)cc(C)sn1 C(c1ccc2ncccc2c1)=CC(=O)NC(C(=O)OC)CC1CCCCC1 C1(NC(=O)CCCCC2CC2)CN(C(c2ccc(F)c(F)c2)=O)CC1C1CC1 NS(=O)(=O)C1(C(=O)NC2CC(F)(CNC(C3(C(F)F)CC3)=O)C2)CCC1 c1(CC2C(C(=O)NC(c3cn(C(C)(C)C(=O)O)nn3)C)C2)ccccc1 N1(C(=O)OC(C)(C)C)CCC(CNc2nc(-c3ccccc3)cs2)C(C2CC2)C1 c1(C(=O)NCCCCCCNC(C2C(C)(C)C2(C)C)=O)ccn2c1CSCC2 c1(CC(=O)NC2CC(C)(NC(C(C(C)C)c3ccccc3)=O)C2)ccccc1C#N CCC(CC)(CN=c1nc(N(CC(C)(CC)OC)C)c2c([nH]1)CSC2)C(C)C c1(NCCCc2n[nH]c(=N)s2)cc(S(=O)(=O)NC(c2ncccn2)C)ccc1C#N C1(C(CC)CNC(=O)C(N)=O)CCN(C(=O)CN(C2CCC2)C)CC1 C1(NC(CCCOCC)=O)CCCN(C(=O)C(C)=C2CCCC2)CC1F C1(C(=O)NC(C2CCCN2C(=O)Cn2cnc(Br)n2)(C)C)CCC(=O)N1 N1(C(Cc2c(OCC)cccc2)=O)CCC(NC(C2COC2)=O)C12CCCC2 O=C(CC1=Cc2ccccc2C1)NCCn1cc(CC(c2ccccc2)O)nn1 N1(C(C(CC(C)(C)C)O)=O)CC2CN(C(c3cccnc3O)=O)CC2(C)C1 C#Cc1cc(C(N2CCN(C(c3csc(C)c3)=O)C(C)C2)=O)cc(N)c1 CC(CCOC1CC1)N=c1nc2c(ncn2C)c(NCCCN(C)C)[nH]1 c1(N)cnccc1.N1(C(C2(CC)CC2)=O)CCC(N2CCN(C3CC3)CC2)CC1 N1(C(C)=O)CCC(C)(C(N2CCOC(C3CN(C(=O)CC4COCCO4)C3)C2)=O)C1 CC1CCCN(C(C2CC2(C)Br)=O)C1CNC(C12CCC(C(N)=O)(CC1)C2)=O N1(C(CNC(=O)NC)=O)CCCC(C)(C)C1CNC(=O)CC1CCC(C)(C)CO1 C1(OCC(C)C)CC(NC(c2cnccn2)=O)C1(C)C c1(CC)ccc(SC(C)(C)C)cc1.N12CCCC(C1)CCOC(=O)CCC2 C1(c2cccc(C)n2)NC(=O)N(c2ccc(F)cc2)C2=C1C(=O)N(C(C)C)CC2 Cc1cc(C(=O)NC(CNC(c2cnc(-c3ccsc3)s2)=O)CO)c(C)cn1 N1(C(COCCC(C)C)=O)CCOCC1C(=O)NC(c1ncn(C)n1)C c1(CC(=O)N(CCCNC(C2CC2F)=O)CC)cc(F)c(Br)cc1[N+](=O)[O-] N1(C(c2ccc(OC)cc2)=O)CC2C3CCC(C2C1)N(C(c1csnc1C)=O)C3 N1(C(C2C(NC(C3(CC)CCCO3)=O)CCCCC2)=O)CCC(O)CC(C)(C)C1 N1(C(c2c(C)oc(Cl)n2)=O)CCC2CN(C(c3sc4nccn4c3C)=O)CC2C1 C(CC(CC)C(=O)N(CC(C)C(=O)NCc1nccc(OC)c1F)C)=CC C(=O)(C(O)C(C)(C)CC)NCCC1CN(C(C2(CC#C)CC2)=O)CC1C N1(C(c2ccc(OC)cc2)C(=O)NCCCCCC)CC(O)C(C)(C)C1 C1(CCOC)(CC)CN(C(C2CC2C(C)(F)F)=O)C1.C1CCC(=O)CNC(=O)N1 C12(C(=O)NC(C)Cc3ccsc3)CC(COC)(CN1C(=O)C(O)c1ccsc1)C2 N1(C(c2c(C)ncnc2)C(=O)NCCOC2CC2)CCC(C)(C)C(CO)C1 CCCS(=O)(=O)CC(=O)N1CCC(N(C)C(c2cnc(C(C)O)s2)=O)C1 N1(CCNC(C2CN(c3ncccn3)CCC2(F)F)=O)Cc2ccccc2C1 C(=O)(N=c1ccn(CC(C)C)[nH]1)C12CCC(NC(C=CC(CC)C)=O)(CC1)C2 C1(CCC)CN(C(=O)COCCCOC)CCN1C(=O)CCC1CCCCN1C CCC(C)(C)C(C)NC(=O)CC1(C)CCN1C(=O)CC(CC)C1CC1 c1(C(N(CC(CNC(C(C)OCCCC)=O)(C)C)C)=O)cc2c(F)cccc2[nH]1 N1(C(CC2CCCC(OC)C2)=O)CC(C)(C)CC1C(=O)NC1CC12CC(O)C2 CC1CC2CC2CC1C(N1CC(CNC(=O)CN2CCOC2=O)C1)=O C(CC(C(=O)N(C)Cc1cnnn1C)NC(=O)CCCC#N)N(C)C c1(N(c2ncc(O)cn2)C(C2CCC(C(C)C)NC2=O)=O)ccc2c(c1)CCNC2 C1(CC)C(NC(c2ccc(OC)s2)=O)CCCN1C(=O)CCC1CCOC1 c1(CCC(=O)Nc2c(OCCN(C)C)cccc2Cl)cnc2c(Br)cccn12 Cc1ccc(OC(C)C(=O)N2CC(CCNC(C34COC(C)C3C4)=O)C2)cc1 C1(C(=O)NC2C(CNC(c3cnc(-c4ccccc4)[nH]3)=O)C2)CCCC1O c1(SCC=C)ccc(C(=O)NCC23CC(NC(C4CC4=C)=O)(C2)C3)cc1 CC1C(c2cccc(F)c2)OCCN1C(c1ccc(F)c(Br)c1)C(=O)O N1(C(c2n(C(C)C)ccc2)=O)CC2(CNC(C3COC(=O)N3C)=O)CCC1C2 Cc1nc(N2CCCC2CNC(=O)CC2CCC(C)C(C)C2)cc(Cl)n1 N1(C(C(C)N(C(C)=O)C)=O)CCC2(CCCC2CNC(c2cnco2)=O)CC1 CC1CN(C(c2cnc(NC3CCOC3)s2)=O)CCN1C(=O)CC1CCCCC1 CC1(CC(=O)NC2CC2CNC(=O)C(c2ccc(Cl)nc2)(C)C)CCS(=O)(=O)N1 CCCCCCC(F)C(=O)N1CCC(CCC(C)(C)NC(=O)C=CCO)CC1 CC(C)CC(O)C(=O)N1CCC(C2CCCN2C(=O)CC2COC(=O)C2)C1 c1(C(=O)NCC2CN(C(CC(COC)(C)C)=O)CC2C)c[nH]c2cc(Cl)ccc12 N1(C(C(C#N)=CC(C)C)=O)CCC(C)C(NC(C2CCC(N=[N+]=[N-])C2)=O)C1 C1(CNC(c2c(C)snc2)=O)CN(c2ncc(C#N)cc2Br)CC12CCOCC2 C=CCC(C(=O)NOCCCOC)NC(=O)CCCN(C)C c1(CNC(C2CCCN(CCC(=O)OC)C2)=O)noc2ccccc12 Cc1ccc(F)c(C(N2CC3CC(NC(=O)Cn4nccn4)CC3C2)=O)c1N c1(C(=O)NC2C(C)CCN(C(c3ncccn3)=O)C2)cccc2c1CCC2 C1(CNC(C(C(C)C)SC)=O)CC(C(C)(C)C)CCN1C(c1cscc1F)=O N1(C(c2ccc(CCC)[nH]2)=O)CCCC(CO)(CNC(=O)CCC2CC2C)C1 c1(CC(N2CC(CC=C)(NC(C3(F)CCOC3C)=O)C2)=O)ccc2c(c1)OCO2 C1(CNC(c2n(C(C)C)ncc2)=O)CCC(C)N(C(c2cc(CCO)on2)=O)C1 C(=O)(C1=C(C)OCCC1)NC(CC)CNC(c1cncc(C(N)=O)c1)=O c1(C(=O)NC(C)CCCNC(=O)C2=CCCCO2)cc2c(Br)cccc2[nH]1 Cc1ccc2[nH]c(C(N3CC4CC3CCC4NC(=O)C(C)O)=O)c(C)c2c1 Cc1nccc(C(=O)NC2CC(F)(F)CC2NC(=O)C(C)CCN(C)C)c1C C1(CNC(C2CC(=O)NC2)=O)(NC(C2(C(F)(F)F)CC2)=O)CC2CCC1CC2 c1(CC)noc(CC)c1CC(=O)NCC1C2CN(C(=O)C3=CCCC3)CC12 C(C(=O)NOC1CCCCC1)C1(CNC(CN(C)C)=O)CC1 CCC(CC(=O)NCC1(O)CCN(C(=O)CCCC(OOC)CC)C1)C(C)(C)C N1(C(C2(CC)COC2)=O)CC2COCC2(C(=O)NCCCCC(C)(C)C)C1 CC1CN(C(C2CCS2(=O)=O)=O)CCC1C(=O)NC(C)C(C)(C)CO N1(C(CCN(CC)CC)=O)CCCC(CCNC(c2ccncc2C(F)F)=O)C1 C1(NC(C(CC#C)C2CC2)=O)(CC)CCN(C(=O)CN(CC(=O)NC)C)CC1 N1(C(c2ccc(CC)cc2Cl)=O)CC2CC(C1)CN(C(=O)C(C(C)CC)OC)C2 C12CC(C(F)(F)F)CCN1C(=O)N2.c1(C(C)(C)C)nnn(CCc2nnnn2C)n1 c1(C(=O)NC(C)CCCNC(=O)C2=CCCOC2)c(O)cc(=O)n2c1CCCC2 Cc1cc(C(N2CCC3(NC(=O)Cc4csnc4C)CC3C2)=O)c(Cl)cn1 C12(NC(C3CCC(NC(CC4(C)CCOCC4)=O)C3)=O)CCCC1C2(F)F N1(C(C(C)SCC)=O)CCCC(C(=O)NCc2cc(OC)ccc2F)CC1 C(C(C)(O)CCO)NC(C1C(NC(C2(CC=C)CCCC2)=O)CC1)=O C=C1CC2(C1)CN(C(=O)CCC(C)NC(=O)C(C1CCOCC1)C)C2 C1(CC(=O)NC(c2ncc[nH]2)CC)CCCN(C(C2CC(O)CN2C)=O)CC1 C=CCCCC(C)(C)C(=O)NCCC1CN(C(=O)Cc2cc(C)[nH]n2)CCO1 Cc1cncc(CCC(=O)NC2CCC(CNC(=O)Cc3n[nH]c(C)n3)CC2)c1 C(=O)(C(O)C1=CCCCC1)NCC(CNC(C1CNC(=O)N1)=O)OC C1(NC(C2C(C)(C)COC2)=O)CCCN(C2CCCc3ccc(F)cc32)C1 N1(C(CCC#C)=O)CCC2CCN(C(=O)CCC(=O)NN(C)C)C2C1 CC1CCOCC1C(=O)NCC1(O)CC(C(=O)NC(c2nn(C)cc2O)C)C1 N#CC1CN(CCN2CCCC2)CC1NC(=O)CC(O)c1ccccc1 c1(-c2nccc(C(=O)NCc3ccnc4[nH]ccc34)c2)c[nH]c2cnccc12 c1(C(=O)NC(CN(C(C=C(COC)C)=O)C)C)nc(C)c(C)nc1O C1(CNC(CC(C)N)=O)CCN(C(=O)C(=O)NC2CC2)C12CC2.C(N)(=O)NC(N)=O CCC(CC)(CCO)CN=c1ccc(Br)c(S(=O)(=O)NC2CC2(C)C(C)C)[nH]1 C1(NC(CC2C(C)CCO2)=O)CCC2CCN(C(=O)CCC3CC3(Cl)Cl)C1C2 C1(CNC(C2(CC=C)CCN(C(=O)CC3CCOC3)C2)=O)CCC2(CCC2)O1 c1(SC)ccc(C(=O)NC(C)C(c2cccc(C)n2)C)cc1Br C1(C(=O)NCC(CO)NC(c2ncc(C)nc2)=O)Cc2ccccc2C(=O)O1 N1(C(c2cc(C)sc2)=O)CC(CNC(=O)Cn2cnc([N+](=O)[O-])n2)CC(C)(C)C1 C(C1COc2ccccc21)c1nc(CCCCC)n(-c2ccn(CCC)n2)n1 C1(C(=O)NCC2(CCC)CCC2)(CNC(=O)CC2OCCCO2)CC2(CC2)C1 C(c1ccccc1F)=CCC(N1C(CNC(C2C(COC)C2)=O)COCC1)=O C=CCC(CC)C(=O)N1CCCC1C(C)(C)NC(c1c(C)noc1C)=O CC(C)(O)C(C(=O)NCCCS(N)(=O)=O)NC(=O)CCC1OCCO1 c1(C(N2C(C)C3CC2C3NC(C2CC(=O)N(C)C2)=O)=O)c[nH]c2ccc(F)cc12 C1(CNC(C2CC(OC)C2)=O)CC(F)CN1C(=O)CCc1csnn1 c1(NC=O)ccc(F)c(CC(=O)NC2CC2CNC(C23COCC2C3)=O)c1 S(=O)(=O)(c1cccc(C(N2CCCC(CNC(=O)C(C)N(C)C)CC2)=O)c1)NC Cc1ccnc(C(=O)NCCN(C2CCCC2)C(c2c(C)ncnc2C)=O)c1N CC(C)CCCC(C)C(=O)N1C2CCC(C(=O)NCC34CC(CCO3)C4)C1CC2 Cc1c(C(N2CC(NC(C34CC5CC3C4C5)=O)CC23CCC3)=O)cccc1C#N N1(C(CCC(C)OCC)=O)CC2(CCN2C(=O)Cc2ccoc2)C1 c1(C(N2CC3C(NC(=O)Cc4csc(Cl)n4)(CC3)C2)=O)ccc([N+](=O)[O-])cc1 C1(CNC(c2ccc(COC)cc2)=O)CCC(C)CN1C(=O)CC(F)(F)F C12CC(C1(C)C)CNC(=O)CN2.c1(C(=O)NCCNC(C)=O)cscn1 N1(C(=O)NCc2n(C)ncn2)CC2CS(=O)(=O)CC2C1 N1(CCC(=O)N)C(=O)CCC1=O.Cc1noc(CCC(=O)N(C)CC2(C)CC2)n1 C1(NC(C2N(C(C)=O)CCCC2)=O)CCC2CC1CN2C(=O)C(N)=O c1(OC)ccc2c(c1)CC(C(=O)NC1(CNC(=O)COC3CCCOC3)CC1)O2 c1(C(=O)NCCCCCC(=O)NC(CCOCC)C)ccc(C#N)c(C)c1 C1(N(c2cn(C)nc2)C(C2CC2(c2ccc(F)cc2)C)=O)CCNCC12CC2 C(=O)(C(O)C(F)(F)F)NCC(C)(CO)NC(c1c(C)[nH]c(-c2ccccc2)c1)=O N1(C(C2C(C)CC2)=O)CC2(C)CC1(C(=O)NCC(C)(C)C#N)C2 CCC(C)C(C(=O)N1CCCC1(C)C(=O)NOCc1ccc(O)cc1)OC N1(C(CCOCCOCC)=O)CC(NC(C2CN3CCC2C3)=O)CC(C)(C)C1 C1(C(N(CCNC(CC(CC)OC)=O)C(C)C)=O)CCc2nn[nH]c2C1 c1(C(N2CC(CC(C)NC(=O)Cc3c[nH]nc3O)C2)=O)ncoc1C(C)(C)C Cc1nc(C(=O)NCC2CCN(C(c3ccoc3Br)=O)C2)c(=O)[nH]c1C C1(N(C(CCN(CCC)C)=O)C)CCN(C(=O)CCc2cc(C)no2)C1 Cc1cnc(C(=O)NCC2CC(O)CN2C(C2CCN(CC(C)C)CC2)=O)nc1 C1(NC(CC(C)OC)=O)CCC2(CC1)CC(NC(c1ccc(F)c(F)c1F)=O)C2 C1(CNC(C(=O)NCC#C)=O)CC2CCC1N(C(=O)CCCCCCC)C2 Cc1ccc2[nH]c(C(N3CC4CC(NC(C5CCCS5)=O)C3C4)=O)cc(=O)c2c1 N1(C(C(C)OCC=C)=O)CC2(CCC(NC(=O)C(C)Cc3ccco3)CC2)C1 c1(OC)ccnc(C(N2CCC(OCCNC(C3(Cl)CC3(F)F)=O)C2)=O)c1 c1(C(N2CCN(C(=O)Cn3cnc(Br)c3)C(CO)C2)=O)cccc2[nH]ccc12 C#CCCCC(=O)N1CCCCC1C1(NC(=O)C=CC=C(Cl)Cl)CC1 N1(C(CC2(C(=O)OC)CCOCC2)=O)CC=C(CNC(=O)Cc2c[nH]nc2O)CC1 Cn1ncc(C2CC2)c1C(N1CCOC(CNC(=O)C(F)CC2CCOC2)C1)=O N1(C(CC2C(C)(C)CC2)=O)CCN(C(=O)C(c2cccc(Cl)c2)(C)C)CC1CO C(=O)(C(=O)N=S(C)(C)=O)NCCN(C(C=Cc1n(CC)ncc1)=O)CC1CC1 C1(CC)CN(C(c2c(OC)cccc2F)=O)CCN1C=O.C1(OC(F)F)COC(=O)C1 Cc1cccc2c1OC(C(=O)NCC1CC(NC(=O)Cn3ncn(C)c3=O)C1)C2 N1(C(CC(CC)CC)=O)CC(NC(C2CCC=CO2)=O)C2CCCCC12 C(=O)(C(F)C(F)(F)F)N(C(C)(C(=O)N(C1CCCC1)C)C1CC1)C N1(C(c2cc(C)nc(C(F)(F)F)n2)=O)CCC2CN(C(=O)CCF)CCC12 C1(O)(C(N2CCC(C(C)NC(C3(OCC)CCCC3)=O)C2)=O)CC(C)(C)C1 C1(C(=O)NC2(CNC(c3ccsc3Br)=O)CC2)CC12CC2(F)F N1(C(C(CC)CC2CCCC2)=O)CCN(C(C)=O)C(c2c(C(C)=O)csc2C)C1 CC(C)(CNC(=O)CC1CCC(=O)N1)CNC(C1(n2cccc2)CCCC1)=O C1(CN(C(=O)CCC2CCCCO2)C)CCN(C(=O)CSCC2CCCO2)CC1 c1(OC)cc(F)c(-c2ccc(CNC(c3cccc(Cl)c3)=O)cn2)cc1F N1(C(c2cc(CC)no2)=O)CC=C(CC(=O)NCCCc2nncs2)CC1 C1(CC)CCCC(C(=O)O)N1C(c1ccc(-c2ccccn2)nc1)=O CCS(=O)(=O)C1CN(C(=O)CC2CCN(C(c3cccc(COC)c3)=O)C2)C1 C(=O)(C(CC(F)(F)F)c1ccc(O)cc1)NCC(=O)NC1CCN(C2CC2)CC1 c1(CNS2=CC=CC=C2c2cc(NCCCCCCCCO)ccn2)ccn2ccccc12 c1(C(N2CCC(C#N)(N)C2)=O)ccc2nc(O)oc2c1.CC1=CCC(C(=O)N)CC1 N(C=CC(=O)C(F)(F)F)C(=O)NCC1CCC(N(C)C)C1 C1(NC(C2(OC)CCC2)=O)CN(C(c2cncc(F)c2)=O)CC1n1cccn1 N1(C(C=CCOC)=O)CCC(NC(C2CC(=O)N(c3ccccc3)C2)=O)C(O)C1 C(=O)(C(C(C)(C)O)NC(=O)CCC1CCOCC1)N1CCCC(OC)C1 c1(-c2c(COC)cccc2)cccc2[nH]c(C(=O)Nc3cc(O)ccn3)cc12 Cc1cn2cc(CC(=O)Nc3cnn(-c4ccc(F)cc4)c3)nc2s1 O=C(C#CC1CCOC1)NC(CCF)C(=O)NCc1nncs1 N1(C(=O)CCn2cc(CN3CCCC3=O)nn2)CC2(CCOCC2)C1C1CC1 C(=O)(C(O)CC(N)=O)N(CCC)CCc1cnn(C)c1CC(C)C.C(C)(=O)O c1(C(N2C(CN(C(C(CCC#C)O)=O)C)CC(F)C2)=O)ccc2c(c1)OCCO2 C1(CNC(C2(CC=C)CCCN2C(c2oncc2CC)=O)=O)C2CCCCCC12 C1(NCC2(CCC=C)CC2)CCC(NC(=O)C(O)CO)CC1 C1(C(=O)NC2CCN(C(c3[nH]c(CC)c(Cl)n3)=O)CC2)CC1C1CCCC1 N1(C(=O)COCc2cccnc2)CCN(C(C2CC23CCC3)=O)C(C2CCC2)C1 N1(C(CC(=O)NCC#C)=O)CC(F)(F)CC1CNC(c1cccc(CCO)c1)=O Cc1csc(C(=O)NCC(C)NC(c2c(C)n[nH]c2C)=O)c1Br c1(C(N(C)C)=O)cccc(-c2cscc2C(=O)NC2CC(O)C2)c1 S(=O)(=O)(c1ccc(Cl)cc1)N1CCCC(N(CCN2CC(=O)N(C)C2=O)CC)C1 N1(C(C(c2ccccc2)=O)=O)CC2CC1C2NC(=O)C=CC1CCOCC1 N1(C(=O)NCc2ncnc(O)c2F)CCc2ccc(Cl)cc2CC1 Cc1cc(N)ccc1C(=O)NCCC1(CNC(=O)Cc2ccnn2C)CC1 c1(C(=O)NC2CCCN(C(CC3CCCC(C)O3)=O)C2)ccc(F)c(F)c1 N1(C(c2nccc(OC)c2)=O)CC(NC(=O)C(C)(C)CO)CC(O)C1 c1(C(N2CC(O)(CNC(C3C(C)(C(F)F)C3)=O)C2)=O)cc(O)nc(O)n1 c1(CNC(CCNC(C(c2ccnn2C)C)=O)=O)cc2cc[nH]c2cn1 CCCCCCC(F)C(=O)NCCC1(O)CN(C(C2(c3ccnn3C)CC2)=O)C1 C(=O)(C1=CC2(CN(C(c3ccncc3)=O)C2)OC1)N1CCC(C)(F)C1 C1(C#N)(CC(N2C(CC(=O)N(C)CC3CC(O)C3)CCCC2)=O)CCOCC1 n1(CC(N2CCC(OCCNC(C3(O)CCOC3)=O)C2)=O)ccccc1=O c1(C(N2CCC(C3CCCCN3C(=O)C3CC3)CC2)=O)c(F)ccc(Cl)c1F Cc1sc2ccccc2c1C(N1CC2CC(NC(C3C4CCCC34)=O)C2C1)=O C12(NC(=O)C(O)Cc3cnc[nH]3)CCC(CC1NC(C1(N3CCCC3)CC1)=O)C2 n1(C(C)C)cc(C(=O)NC(C)C(C)NC(c2sccc2OC(F)F)=O)cn1 C(=O)(CC(C)(C(F)F)N(C)C)NC(C)CNC(c1cc(C2CC2)cs1)=O c1(C(=O)NCC2N(C(C3CC(OCC)C3)=O)CC(CO)C2)c(F)ccc(OC)c1F C1(CN(C(C2N(CC)CCC2)=O)CC)CCN(C(=O)Cc2nncn2CC)CC1 C(=O)(C(F)CC1CCCC1)NCCOCCCNC(=O)CO N1(C(C(CC)NC(N)=O)=O)CC2(C=C(C(=O)N3CCOCC3C)CO2)C1 C1(C(=O)NC(CC)=O)COCCN(C(=O)C(C)C)C1 CC1OCCN(C(=O)C=CCN(C)C(C2CCC(=O)N2C)=O)C1CN(C)C CC1CCCC(C(N2CC(O)(C(F)C(=O)NCCn3ccc(=O)cc3)C2)=O)CC1 N1(C(C2C(C)C2)=O)CCN(C(c2cnc(Cl)s2)=O)CC1c1cccc(F)c1 C1(CNC(C=CCOC)=O)C2CC2CN1C(c1conc1C(F)(F)F)=O N1(S(C)(=O)=O)CC2CC2C1.c1(C(N2CC(=O)NCC2)=O)cnc(Cl)s1 c1(C(=O)NC(CN(C(=O)C=Cc2cncn2C)CC)C)nc(Br)cnc1N C(CC(F)F)(C(=O)N1CCC(CC2CC2)C1)N(C(c1ccc(C2C(C)C2)o1)=O)C Cc1nc(C(=O)NCC2(NC(=O)C=Cc3ccnn3C)CCC2)nn1C c1(-c2n(CCC(=O)OCC)nc(C(CC)CC)n2)ccc(C)n(C)c1=O C(=O)(C1=NNC(=O)CC1)NC1CC(C)N(C(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C1 CC1CC(CCNC(=O)C2CC2)CCN1C(c1cn(C)nc1-c1ccoc1)=O C1(CC(C)NC(CN(CCOC)C)=O)CCN(C(=O)C(C)C2CC2)CC1 Cn1cncc1C(N1CC(NC(C2CCCC2n2cccc2)=O)C1)=O Cc1cc(F)c(CNC2CCCC2C(=O)Nc2cscn2)c(F)c1 Cc1[nH]nc2ncc(C(N3CCN(C(=O)Cc4nc[nH]n4)C(C(C)C)C3)=O)cc12 c1(C(C(=O)NC(C)(C)C)N(C(C2(C)CC2)C)C)ccnc(Cl)c1OC CC1=CC2CC(C1)CC(c1nnnn1Cc1cccs1)(Nc1csnc1C)C2 c1(C(=O)NC2C3CN(C(c4cc(CC)c(CC)o4)=O)C2C3)cncn(C)c1=O C(=O)(C(C)(C)CC(F)(F)F)N1CC(C)C(NC(C2CNC(=O)C2)=O)C1 Cc1ccsc1C=CC(N1CCOC(CNC(=O)CCSc2ccccc2)C1)=O C12(CCC1)C(=O)NCCN(CCOCC)C2=O.C1(C)(SC)CC1 C(c1cncnc1O)=CC(=O)NCC1CCCN1C(c1n[nH]cc1Br)=O C1(c2n(CCC)cnc2)NC(=S)N(CC(C)C)C(C2CCC2)=C1C(=O)OCC Cc1ccc(C)c(CC(=O)NCC2CCC2NC(=O)CCNC2CCCCC2)c1 c12cccc(c1)C(=O)N2.c1(CCOCC)cn(CCN(CCCCO)C)nn1 c1(C(N2CCC(NC(CC3ON=C(C)C3)=O)CC2)=O)nccc(F)c1Cl C1(C(=O)NCC(C)N(C(=O)CCN2CCCCC2)C)CCCCC12CCC2 c1(C(=O)NC(CCN(C(c2c(C)cccc2Cl)=O)C)C)cccc2nc(O)oc12 c1(CC)cccnc1C(=O)NCCC1CCC(NC(=O)CO)C1 C#CC1(C(=O)NC2(c3ccccc3)CN(C(=O)CNc3cnoc3C)C2)CCCC1 C=C=C(C)CC(=O)NCCC(C)CCNC(c1ccn(C2CCCCC2)n1)=O c1(CC(C)(C)OC(C)=O)cn(CC(C)NC(=O)C(F)(F)C2CCCC2)nn1 C(C)(C)(C(=O)NCC1(O)CN(C(=O)CCNC(c2cccn2C)=O)C1)OC(C)C CS(=O)(=O)CCN=c1[nH]c2c(c(=NCCOCCS(C)(=O)=O)[nH]1)CCCC2 CC1(CNC(=O)COCCc2ccccc2)CCN(C(c2cncs2)=O)CC1 CC(N=c1cc[nH]c2ccc(C(F)(F)F)cc12)C(=O)OC(C)(C)C C1(C(=O)NCC2CCN(C(c3ccc(SCCC)cc3)=O)C2)CC(C2CC2)=NO1 Cc1nnc(O)c(C(=O)NCCC2(CNC(C3(C)CCCOC3)=O)CC2)c1C c1(OC)ncnc(CNC(=O)Nc2cc(C(F)(F)F)cnc2O)c1Cl C1(NC(C(C(C)C)OCC)=O)CC2CCC(C1)N2C(C1CC1C(F)(F)F)=O N1(C(C=CCN(C)C(C2SCCS2)=O)=O)CC2CC=CC1C2 C1(CNC(c2c(C)ccnc2)=O)CN(C(=O)C(CO)C(C)C)CCC12CCOC2 CC(=O)CCCC(=O)NCCC(C)NC(=O)CC1CCCC(F)(F)C1 c1(C(=O)NC2C(C(=O)NC(CCC(=O)OC)C)CCC2)cccc(C(F)(F)F)c1O C#Cc1cccc(C(=O)NCC2CN(C(c3cc(OC)cs3)=O)CCC2C)c1C C(C(=O)N=c1ccn(C2CCOC2)[nH]1)(c1cc(F)ccc1Cl)OC c1(CC)ccsc1C(N1CCCC1C(C)(C)C(=O)NCc1cc(C(N)=O)no1)=O n1(CC(CC)O)cc(C(N2CC(O)(CNC(=O)CCN3CCC3)C2)=O)nn1 c1(NCC(CSC)OC)ccc(S(=O)(=O)NC2CCOCC2OC)c(Cl)c1 N1(C(c2n[nH]c(C)c2C)=O)CCN(C(c2ccc(-c3cscn3)cc2)=O)CC1C N1(C(CC(CC)N(C(=O)CC2CCCCN2C)C)=O)Cc2cnn(C)c2C1 c1(OC)ncccc1C(=O)NCC1(CNC(C2C(CO)C2)=O)CC12CCC2 Cc1c(C(N2CCOCC(NC(c3ccon3)=O)C2)=O)ccc2ccccc12 C(=O)(C1=C(C#N)CCC1)NC1(CNC(C2OCCN(C)C2=O)=O)CCOC1 Cc1cccc(C(F)C(=O)NCC2CN(C(c3c(C)nsc3C)=O)CC2C)c1 C1(NC(c2c(CC)ncs2)=O)CC(CNC(C2(COC)C=CCC2)=O)C(O)C1 c1(C(=O)Nc2cccc(-c3nnc(OCC)s3)c2)c(F)c(C)nc2ncnn12 c1(C(N(CCC(=O)NCC(C)(C)COC)CC#C)=O)sc(C)cc1C Cc1cc(O)ncc1C(=O)NCCCCC1(NC(C2COCCC2C)=O)CC1 C1(C(N(CCCNC(C2(C#N)CCCC2)=O)C)=O)CCCCN1N=O N1(C(C(CO)N(C)C)=O)CC2CN(C(=O)Cc3c[nH]c4ccccc34)CC2(C)C1 S(=O)(=O)(c1cnc(N2CCC3(CCC3)C2)c(Cl)c1)NC(C)Cc1ccco1 C(=O)(CCC(F)(F)F)NC1C(NC(c2cnn(C)c2-n2cnnc2)=O)CCCC1 c1(C(N2C(CNC(CC3CCCC(OC)C3)=O)CC2)=O)ccc(=O)n(CCO)c1 Cc1ccc(C(=O)NCc2ccc(Cl)cc2)c(NC(=O)C=Cc2nc(C)co2)c1 Cc1nc2nc[nH]n2c(=O)c1CCCNC(=O)CC(N)C(F)(F)F c1(C(F)(F)F)nccc(-c2nc(C(F)F)nn2C23CC(C(F)F)(C2)C3)n1 N1(C(C2OCC(C)(C)C2)=O)CC2COCC2(C(=O)NCCc2ncccc2F)C1 N1(C(C(c2cc(C)sc2)(C)C)=O)CCC(CNC(c2ccncc2C)=O)C(C)C1 c1(C(N2CCN(C(C=CCOC)=O)CC2C)=O)cnn(C)c1S(N)(=O)=O N1(S(c2c(C)cccn2)(=O)=O)CCOc2ccncc2C1 CCC(C)(C#N)C(=O)NCC1CC2(CC(NC(=O)CCCCC3CC3)C2)C1 N1(C(c2c(C)[nH][nH]c2=N)=O)CC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 C12(C(=O)NCC#CCNC(C(c3c(C)noc3C)C)=O)CC(CO)(C1)OC2(C)C c1(C(=O)NCC2N(C(C(C)OCOC)=O)CCC2)ccc(C(C)O)cc1 CC(CCCNC(c1conc1C(F)(F)F)=O)NC(=O)CCCN1CCCCC1 N1(C(C2C(C)CC2)=O)CC=C(C(=O)NCCCN(C)C2CC2)C1 c1(N2CCC(OC(CF)(F)F)CC2)nc(N2CCCC(O)CC2)nc2c1CCC2 C(=O)(CC(C(F)F)NC(C1(C#N)CCOC1)=O)N1CC(CC(N)=O)C1 N1(C(C(CCOCCO)NC(CN(C)CC)=O)=O)CCC(C)C2(CCC2)C1 C1(CNC(=O)CCC(F)F)CC2CCC1N(C(c1c[nH]c3cccnc13)=O)C2 CCS(=O)(=O)CCNC(N1CCC(N)C1)=O.c12ccc(cc1)o2 CCCC(CCNC(=O)CC1(C)CN(C(c2cccc(OC)c2)=O)C1)CCC Cc1cc(C(=O)NCC=CCNC(C2CCCCS2)=O)nn1CCO C1(C(=O)N(CCCC(=O)N2CCC(n3ccnc3)C2)C)(OCC)CCOC1 N1(C(CCc2onc(CC)n2)=O)CCN(C(c2ccc(O)nc2)=O)CC12CCC2 C(=O)(CS(=O)(=O)CC(C)C)N1CC(CNC(c2c(Cl)ccc(C)c2N)=O)C1 C12(C(N(CCCC)CC)=O)CC(CN1C(c1cccc(C)c1)=O)C2 Cc1cc(-c2ccc(NC(=O)CC(C)N(CCC#N)C)cc2)cc([N+](=O)[O-])c1O C=C(CNC(c1cc(C)cs1)=O)CCNC(C1CCCN1NS(C)(=O)=O)=O Cc1ccccc1C(=O)N(C)CCNC(=O)Cn1ncn(C)c1=O C1(C(=O)NC2(CN(C)C(c3ccc(Br)[nH]3)=O)CC2)CCn2cnnc2C1 N1(C(CC(CC)C2CCC2)=O)CC(CNC(=O)C(C)=C2CCC2)CC12CCC2 N1(C(c2ccnc(OC)c2F)C(=O)NCCCSC)CCN(C(C)=O)CC12CC2 NC(=O)CCCCC(=O)N1CCCN(C(=O)COCc2cccc(Br)c2)CC1 c1(-c2cnc(C(C)NC)s2)nc(-c2ccc(OC)cn2)nn1C(C)C(C)C c1(CC(=O)N(CCCOCCN(C(CCC)=O)C)C)c(F)cc(F)cc1F Cc1c(CNC(N2CC(C)(C)CC2c2ccc(F)cc2)=O)ccc2nccn12 N12CC(F)(F)CC1CCOC2=O.C1(=C(C)C)CCN(C(C(C)(C)C)=O)C1 c1(C(=O)NC(C2OCCN(C(c3ccc(OC)s3)=O)C2)C)cc2cccnn2c1 c1(NC(c2ccc(C#C)o2)=O)cc(OC)c(OC)cc1OC CC1COC2(C1)CN(C(C1CC3CCC1N3C(C1CCSC1)=O)=O)C2 Cc1cc(Cl)c(C(N2CCC(CNC(c3cnc(C)n3C)=O)C2)=O)cn1 C(=O)(C#CC1CCOCC1)NC1C(NC(c2c(OC)scc2)=O)CC1 N1(C(c2c(CNC(Cc3c(C)scc3)=O)nccc2)=O)Cc2cnn(C)c2C1 CCCCC(CN=c1[nH]cnc(Cl)c1C(=O)OC)NC(=O)C(C)(C)CO Cn1nnc2cc(C(=O)NC3(CNC(C4(F)CCOC4)=O)CCCCC3)cnc12 c1(SCC(=O)NCC2(CNC(c3cc(C)ns3)=O)CCC2)ccccc1Br C(C)(C)(CCC(=O)NC(c1cc[nH]n1)C)NC(C(C)SC(C)C)=O c1(NC(C2C(C(=O)OC)COC2)=O)oc(CNC(=O)C=CC(C)(C)SC)nc1C CCC(CC(=O)N1CCCC1(C)C(=O)NCC1(CC2CCC2)CC1)C(F)F c1(C2C(C(N=c3[nH]nc(CCCC)s3)=O)C2)cc(F)cc(F)c1OC c1(N2C(C)(C)C(NC(C3CC4C(C3)C4(C)C)=O)CC2)nc2cc(F)ccc2o1 CC1CCCCC1(CNC(c1n[nH]c(=N)s1)=O)NC(C1CCC(C)CC1)=O c1(C(=O)NC)ccc(OC)c(-c2ccc(CNC(c3ccc(Br)nc3)=O)cn2)c1 O=C(CC(F)(F)Cl)NCC1CC1NC(c1nc[nH]c1C(F)(F)F)=O CCC(CCO)C(C)NC(=O)C(=O)NC1COC1 C(C)(CCCCNC(=O)C=CC(C)C)NC(CCSCC(C)C)=O c1(CCNC(N2CCCC(C(C)N)C2)=O)ncc(F)cc1F c1(C(OC)OC)cccc(CN2CCC(O)C2C)c1 N1(C(c2nc(CC)oc2)=O)CCC2C(C1)NC(=O)CCN2C(=O)Cc1ccon1 C(CC(=O)NCCCNC(=O)Cc1ccon1)N.C1(OC(=O)NC)(C)CC1 C1(C(N(C(CCCCC)C2CCC2)C2CCN(C)CC2)=O)Cc2ccccc2C1 N1(C(C(C(=O)OC)C)=O)CC2CN(C(=O)Cc3cc(C)nn3C)C2C1 C1(C(N2CCCC(C(=O)O)(CO)C2)=O)COCC2(CCNCC2)O1 c1(C(N2CCC(O)(C(=O)OC)C2)=O)c(F)cccc1Br N1(C(C)=O)CCC(CC(=O)NCC23CC2CN(C(=O)C=CSC)C3)CC1 CCCC(F)(F)C(=O)NCC1CCCC1NC(=O)CC1CCCCC1O c1(C(=O)NCCCNC(C2(C)CC2F)=O)cnc2cnc(Cl)cc2c1 C(=O)(C1=CCCCCC1)N1CC2(CN(C(CCCc3ncc(C)o3)=O)C2)C1 N1(C(c2nccc(C)n2)=O)CCN(C(C2CC2F)=O)CC1CC#N c1(C(c2nnnn2CC2CC2)NC(c2cnn[nH]2)C)cc(I)n(C)n1 C12(NC(CC(COC)C)=O)CCCC1CN(C(c1ncc(N)cc1Cl)=O)C2 c1(C(=O)NCC(C)NC(=O)CN2CC3CC3C2)ccc(S(N)(=O)=O)c(O)c1 N1(C(C(C)OCCOC)=O)CC2(COC(CNC(=O)CCC(C)C)C2)C1 Cc1c(C(N2CCCC(C)(NC(=O)C(C)S(N)(=O)=O)C2)=O)cnn1CCC(C)C C1(O)(C(=O)NCc2cc(C(NOCCOC)=O)no2)CCCCC1 N1(C(CC2COCC(C)O2)=O)CCCN(C(=O)Cn2nnc(=N)[nH]2)CC1 c1(C(=O)NC2CC2CNC(C2(Cl)CC23CCC3)=O)cc2c(Cl)cc(Cl)cc2[nH]1 c1(CCNC(C=C(C)CNC(c2snnc2C2CC2)=O)=O)cccc(F)n1 C(=O)(CS(=O)(=O)C1CC1)NCC1N(C)CCN(C(=O)CCS(C)=O)C1 C(c1sc2ccccc2c1Cl)=CC(=O)NC1C(CNC(C2(O)C(C)(C)C2)=O)CC1 C12(C(N3CC(N(C4CCC4)C(C4C(C)C4)=O)C(F)C3)=O)CC1COC21CCC1 c1(NC(C2CCC(N(C)C)CC2)=O)ccc2c(c1)C(O)CC2(C)C C(=O)(C1=C(SC)CCCC1)NC1COCCN(C(C2C(CC)CC2)=O)C1 c1(C(N(C)CC2N(C(c3cnc(CC)o3)=O)CCC2)=O)ccc(C(C)C)c(F)c1 c1(C(C(=O)NCCCN(C(C2CC(F)C(=O)N2)=O)CC)C)cc(F)cc(F)c1 c1(C(N2CCCC(n3cc(CC#N)nn3)C2)C(=O)NCCC)ncc(Br)c(C)n1 CCCCCCCSc1ccsc1COC c1(C(=O)NCC2CCCN(C(C3CCCC(C)C3)=O)C2)cccc(Br)c1Br N1(C(Cn2nnc(C)n2)=O)CCC2CCCC12CNC(c1scnc1C)=O N1(C(C(C(CC)C)O)=O)CC2(CCC(NC(c3cc(OC)ccc3F)=O)C2)C1 C(=O)(C(C)(C)C1CCN(C(=O)C(Cn2cncn2)N(C)C)C1)N(C(CC)CO)C c1(C(N2CCC(C)(NC(C(C)OCC3CC3)=O)CC2)=O)ccc2c(c1)CCCS2 N1(C(CSCC)=O)CC(CNC(c2csc(C(F)F)c2)=O)C2(CC2)C1 CCCCC(F)C(=O)NC(C(=O)NCCN1CCNC(=O)C1)C(C)(C)O Cc1[nH]nc2ncc(C(=O)NC3CC4CC(C3)N(C(C3(C)CCOC3)=O)C4)cc12 C(CC(C)(CC)NC(c1cccc(Cl)c1)=O)NC(c1ncn(CC)c1)=O N1(C(c2cnc(C)s2)=O)CCN(C)CC1CNC(=O)C(c1ccc(F)cc1)=O CCCCCCCN=c1cc[nH]cc1S(=O)(=O)NCC1C2CCCC12 CON=Cc1ccc(C(=O)NCC2(NC(=O)CC3CCSC3)CCOCC2)cc1 N1(C(C(CCSC)O)=O)CCC(NC(c2cn(C)c(C)n2)=O)C(O)C1 c1(C(=O)NC2(C)CN(C(c3n(CC)c(O)nc3)=O)C2)ccc(OC)cc1F c1(C(N(CC(Cc2ccccc2)NC(C=NOC)=O)C)=O)c(Cl)nn(C)c1Cl N1(C(C2(CCOC)CC2)=O)CC2CCCC(C1)N2C(C1(N(C)C)CCC1)=O C1(N(C(C(CC)O)=O)C)CN(C(=O)CSc2ccccc2F)CC1(C)C C(=O)(C1=NN(C)C(=O)CC1)N1CC2C(CNC(c3c(CC)ccs3)=O)C2C1 C1(O)(CCNC(C2(C)CC=CC2)=O)CCN(C(=O)COc2cccc(F)c2)C1 C1(NC(c2c(C)occ2)=O)CN(C(C2CCCC(C)O2)=O)CC1C(F)F C1(O)(CNC(C(n2cc(-c3cccc(COC)c3)nn2)C)=O)CCN(C)CC1 C(=O)(C(C(C)CC)N1CCCCC1)N1CC(CNC(CC2CC(=C)C2)=O)OCC1 c1(C2(C(N3CC(F)(NCC4CCN(C(=O)C5CC5)C4)C3)=O)CC2)ccccc1F c1(CCC(=O)NCCC(CNC(C2(CC#C)CC2)=O)SC)ccnc(Cl)c1 C1(CC(=O)NCc2c(C)nn[nH]2)CC(C)N(C(C2CCOC2(C)C)=O)C1 c1(C(=O)NCC2C(CC(=O)N(CCCC=C)CC)C2)cc(C)nnc1O C1(C(=O)NCC2CCCCCC2)C2CCC(C2)N1C(=O)COCCN(C)C c1(C(=O)NCCN(C(=O)Cc2csc3cncn23)CC)cc(C#N)c(F)cc1F C1(CC)CN(C(C2CNC(=O)O2)=O)CCC1NC(c1c(C)cnn1CC)=O Cc1n[nH]c(C)c1C(=O)NCC(C1CC1)NC(C1CC1(C)C(F)F)=O N1(C(CNC(c2[nH]cc(C(N)=O)c2)=O)=O)CC2(C1)CN(C(C1CCCO1)=O)C2 C1(NC(C(C(CC)C)OC)=O)CC2(CCC(NC(=O)CCC3CC3)CC2)C1 C1(NC(C2CC3(CCC3)C2)=O)CC2CCC(C1)N2C(C1CCOC1C1CC1)=O C1(NC(C(CCC)O)=O)CCC2CN(C(C3CNc4ccccc4O3)=O)CC2C1 N1(C(c2cnc(OCC)c(Cl)c2)=O)CCCN(C(=O)C(O)C(C)(C)C)CC1CO C(=O)(CC(C(C)OC)SC)OCC.C12(CCOC1)c1c(ccs1)Cn1c2nnn1 Cc1cc(OCc2nc(-c3cncnc3)nn2CC(F)(F)C(F)F)cc(C)c1 N1(C(C(C)C2CCC2)=O)CC2CC(NC(=O)CCc3cncs3)C1C2 C(=O)(C(C#N)C(C)C)NC(CN(C(c1cc(C)[nH]n1)=O)CC)C c1(NC(C2(CC)CN(C(c3cn(CC)nc3)=O)C2)=O)cc(C)cc(C)c1.C1CO1 c1(OC)cc(NC(C2CCC(OC)CC2)=O)c(F)c(OC)c1F c1(C(=O)NCC2(NC(Cc3n(C)cnn3)=O)CC2)cccc2nc(Cl)cn12 N1(C(Cc2n[nH]c(=N)s2)=O)CC2CCC1C(NC(c1nccn3nccc13)=O)C2 N1(C(C(CC=C)(F)F)=O)CCC2(CC1)CC2CNC(=O)Cc1cc(COC)on1 C(=O)(C1=NN(CCO)C(=O)CC1)NCCCN(C(c1cc(C)cc(O)n1)=O)C N1(C(C(CCC)C)=O)CC2CCN(c3nc(C(F)(F)F)c(C)s3)CC2C1 CC1=C(C(=O)NCC(O)CN(C(=O)C(C)(C)c2ccnn2C)C)S(=O)(=O)CCO1 N1(C(C2C(=O)NCC2)=O)CCC2C(CCCN2C(=O)CCc2cccnc2F)C1 N1(C(C(CC)N2CCCC2=O)=O)CC(NC(c2cnc(O)c(O)c2)=O)C(C)(C)C1 C12(NC(C3C4(CC(NC(CCC(C)C)=O)C4)C3)=O)CCC(CC1)C2(C)C c1(CC2CCC(C(N(CC(C)(C)CNC(=O)CO)C)=O)C2)ccc(C#N)cc1 n1(CCOC)nc(C(=O)NC(C)C(C)Nc2nccc(CC#N)n2)ccc1=O Cc1oc(Cl)nc1C(N1CCC(C(C(C)C)NC(=O)COCC(C)(C)C)C1)=O N1(C(C2C(C)(C)C2)=O)CCC(NC(c2cnc(Cl)cc2Cl)=O)C(CO)C1 C=C(C)CC(C(=O)NC1CCC12CN(C(c1cnc(C)cc1Cl)=O)C2)OC N#Cc1ccc(N2CCC(NC(C3CC(c4ccccc4)C3)=O)CC2)nc1 Cc1ccc(C(=O)NC(C2CCCN2C(=O)CC(C)c2ccccc2)C)nn1 Cc1sncc1C(=O)NC1CC1NC(=O)C(C)N1CCC1 c1(C(=O)NCC2CCC(NC(CN(C)CCO)=O)C2)cc(N)ccc1Br c1(C2N(C(=O)Cn3cc(C(C4CC4)Oc4ccccc4)nn3)CC2)cccc(F)c1 c1(C(C)C(=O)NC23CC(CNC(c4coc(Cl)c4)=O)(C2)C3)ccccc1F.C1CC1 C1(C(=O)NC2CCC(NC)C2)CC(O)CN1Cc1ccc(OC)nc1 C=C(C)CC(C(=O)NC(C)(C)C(=O)N(CCC1=CCCCC1)C)OC C1(C(C)NC(c2ccc(SC)s2)=O)CN(C(c2c(Cl)cnn2C)=O)CCO1 N1(C(C(c2ccccc2F)C)=O)CCCC2(CNC(=O)CC(C)(C)C)CCCC12 C(CO)(CC(C)(C)C)NC(CN(C(=O)CC1CSC1)CCC)=O c1(C(N2CCN(C(CC3CCN(C)C(=O)O3)=O)CC2CF)=O)cccc2ccnn12 c1(C(N(CCNC(c2oc(CC)c(C)c2)=O)C2CC2)=O)cc2n(n1)CCCO2 c1(C(N2CC3(CCN(C(C(CC)OC)=O)C3)C2)=O)ccc2ccn(C)c2c1 CC(C)C(C(=O)NCCCC(C)NC(c1c(N(C)C)c[nH]c1C)=O)NC(N)=O c1(C(N2CC(C)C(N(C)C(C3CC(CN(C)C)C3)=O)CC2)=O)cc2ccccc2s1 CCCC(CO)N=c1[nH]c2c(c(=NCC(C)c3ccc(F)c(Cl)c3)[nH]1)CSC2 c1(SCC)cccnc1C(=O)NC12CC(CNC(C3CCCN(C)C3)=O)(C1)C2 c1(C(N2C(CN)CCC(=O)CC2)=O)cc2n(n1)CCCC2 C1(CC(=O)NCC(NOC)=O)CCCN(C(=O)COC(C)=O)CC1 N1(C(c2nc(CC)oc2)=O)CC(C)CN(C(=O)C(C)(C)c2cscn2)CC1C N1(C(CCCN(C)C)=O)CCC2(CC1)CN(C(c1cncs1)=O)CC2CO C(CCCCC(=O)N(C)Cc1nnc(C)s1)N(C(c1c(CC)n[nH]c1)=O)C c1(NC2C(C)(C)CN(C(C34CCCCN3CCC4)=O)C2)ncnc2ccsc12 C(CCCCCCO)NC(c1c(CNC(C2(C)CCCOC2)=O)ocn1)=O c1(CCNC(=O)C(=O)NC2CC2)ccc(F)cc1F.c12ccccc1OC2 C=CCC(CNC(=O)CCC1CC1(F)F)NC(c1cc(OCC)n[nH]1)=O C1(O)(CCNC(C(C)OCCOC)=O)CCN(C(=O)Cn2cnnc2)CC1 N1(C(c2c(C)ncs2)C(=O)NCCC2(C)CC2)CCOc2c(Br)cccc2C1 C(=O)(C(CC(=C)C)NC(=O)C(C)CC=C)N(C(C#C)C)C C1(C(N2CC(C)(NC(C3CCCO3)=O)C2)=O)CCOC1(C)C C(=O)(C#Cc1ccc(Cl)cc1)N1CCC(CC(=O)Nc2scc(C(C)C)n2)C1 C(CC(C)(O)C(=O)NCCCOCCNC(=O)CC1COC(C)(C)CO1)N(C)C c1(C(=O)NCC=CCNC(C(c2c(C)n[nH]c2C)C)=O)cc(F)c(F)cc1F N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)C(=O)NC2CC2)CC1CC(F)(F)F C(=O)(C(CC(C)(C)C)OC(C)=O)N1CC(F)(CN)C1.C1(OC)CCNC1=O.OC Cc1ccn2c(C(N3C4CCC3CN(C(=O)C(C)CN(C)C)CC4)=O)cnc2c1 C(C)C(C)(C)CN(C)C.c1(C(NC)=O)cc[n+]([O-])cc1.CC1CC1=O Cc1c(Nc2ccccc2)ncnc1NC.c1(CC(=O)N)cccc(I)c1F Cc1cc(C(=O)NCCCOCCCNC(=O)CC2(N(C)C)CC2)oc1C c1(C(C)S(N)(=O)=O)ccc(C(=O)N(C)CC2CN(C(c3nc[nH]n3)=O)C2)cc1 C1(N(SCNC(C=CC(=O)CC=C)=O)NC23CC(F)(C2)C3)C2CCC1CNC2 N1(C(c2cccc(C)c2F)=O)CCCN(C(=O)CC2CCCC(C)O2)C(C)C1 CC(C)C(O)C(=O)NCC(C1CCN(C(=O)COC2CCCCCC2)CC1)F c1(C(=O)NCC)cnc2nccc(-c3ccc(-c4ccc(OC)nc4)cc3)c2c1 C1(C(=O)NCC2CCN(C(c3nc(C(C)OC)oc3)=O)CC2)CC2(CCC2O)C1 c1(C(=O)NC(CC)CNC(C2CC=CC2)=O)cc2n(n1)CC(O)CO2 CCC(C)(COC)C(=O)N1CC2CC1CN2C(=O)CCC(=O)c1cc(Cl)sc1Cl C(N=c1[nH]cncc1Cl)c1nc(CNC(CCC2C(C)(C)C2)=O)nc(O)c1 Cc1c(C(N2CCC3C(CCN3C(=O)C(C)CN)C2)=O)cccc1[N+](=O)[O-] C1(C(=O)NCCn2cc(C(=O)NC34CC(C)(C3)C4)nn2)CCCN2CCCC12 S(=O)(=O)(c1cc(Cl)c(F)cc1F)N1C(Nc2ncc(C)s2)CCC1 N1(C(c2c(CC)oc(C)c2)=O)CC(CNC(c2ncccn2)=O)CCC1C n1(CC)nc(C(=O)NC(C)C(C)NC(c2ccc[nH]2)=O)c2ccccc2c1=O CCC(CN(C)C)C(=O)N(CCC(=O)NC(C)CN1CCOCC1)CC Cc1csc(=NCC(=O)NC2CC2CNC(=O)C(c2ccc(C)s2)C)[nH]1 N1(C(c2cc[nH]c2)=O)CCN(C2CCN(C(=O)C(F)(F)c3cscn3)CC2)CC1 c1(C(=O)NC2COCC2CNC(C2CCCCCCC2)=O)cccc2sncc12 C1(NC(C2(CC#C)CCCCO2)=O)COC2(C1)CN(C(=O)CCCC(C)(C)C)C2 N1(C(C(C)SCCCC)=O)CCCOC(CCNC(c2cnc(S)nc2)=O)C1 C12(CNC(C3C(c4ccn(C)n4)C3)=O)CN(C(C34CC(F)C3C4)=O)CC1CCO2 CCC(O)C(C)(C)C(=O)N1CCC(NC(c2ccncc2)=O)C(O)C1 N1(C(c2c(CCC)n[nH]c2)=O)CCC(CF)(NC(c2cc(C)n(CCO)n2)=O)C1 Cc1cc(C(N2CCN(C(c3coc4c3COC4)=O)C(CCO)C2)=O)cc(O)c1 C1(C(=O)NCC2N(C(Cc3c(C)occ3)=O)CCC2C)CCC(C)(C)CC1 N1(C(C2(CCOC)CC2)=O)CCCCC(NC(c2ccc(N(C)C)cc2)=O)CC1 c1(N2CCN(C(c3ccc(C(N)=S)cc3)=O)CC2)cnc2ccccc2c1 Cc1ccc(C=CC(=O)NCCC2(O)CCN(C(c3cocc3C)=O)C2)cn1 C1(CNC(c2cc(F)ccc2O)=O)COCCN(C(C2(O)COC2)=O)C1 CC1COc2c(C(N3CC4(CNC(C5CC(O)C5)=O)CCC3CC4)=O)cccc21 C(=O)(CCC(=O)c1ccc[nH]1)NCC(C)(CNC(=O)CC1CCOC1C)OC S(=O)(=O)(c1cc(C)cc(C)c1)SCC(CC)O C1(CN(C)C(C2CC2Cc2ccccc2)=O)CN(C(=O)CC2(O)CC2)CC12CC2 C12(NC(CCc3ncc(C)[nH]3)=O)CCC(CC1)N(C(c1cc(C(F)F)no1)=O)C2 c1(C(=O)NC2C3CN(C(Cc4cc(C)on4)=O)CC32)ccc(CN(C)C)c(F)c1 N1(C(c2cc(C)n(C)n2)=O)CCC2(CC1)CC(Nc1ncc(C#N)cc1Cl)CO2 C1(C(N2C(c3cn(CCS(C)(=O)=O)nn3)CCC2)=O)CCC2(CCOCC2)C1 N1(C(c2nc(CCC)oc2)=O)CC2CC3CC2C1C3NC(C1CCOC1CC)=O c1(C(N2CC(CC)C(OC)C2)=O)ccc(Br)c(C)c1F CCC(C)C(O)CC(=O)N1CCCC(CNC(=O)CCCNC(=O)C2CC2)C1 C(=O)(C(C(C)C)N1CCCCC1)NC(c1onc(C)n1)C N1(C(c2ccn(C(C)(C)C)n2)=O)CCCC(CNC(=O)CC2CCC(F)(F)C2)C1 C12(C(N3C(C(=O)NCC4(OCC)CC4)C(O)CC3)=O)CCCC1C2(F)F CCC(O)C(C)C(=O)N(CC(C)(C)NC(=O)C(=C1CCCCC1)F)C CC12CC1CN(C(c1ncn(C(C)(C)C)n1)=O)C2 c1(C(=O)O)cc2c(cc1NC(c1ccnn1CC1CCC1)=O)OC(F)(F)O2 c1(C(=O)NCC2N(C(c3c(OC)nsc3OC)=O)CC2)ccc2n[nH]cc2c1Cl c1(OCC)ncccc1N1CCN(C(=O)NNC(=O)C2CC2(F)F)CC1 CC1CCN(C(c2cccnc2F)=O)CC1NC(=O)CCCCCO C1(NC(CCSCC)=O)CCOC(C(N2CCC(C)(O)C2)=O)C1 N1(C(c2c(OC)n[nH]c2)=O)CCC=C(C(=O)NCC23CCCN(CC2)C3)C1 C(CC(C)(C)C(=O)NCC1CC(O)C1)NC(CC(=O)OCC)=O C1(NC(CCNC(=O)CO)=O)CCN(C(c2cc(CO)[nH]n2)=O)C12CCC2 C1(C)(C(N(C2(C(=O)NCC3CCCC34CC4)CC2)C)=O)CC2CCC1C2 c1(C(=O)NC2CN(C(C(CC)NC(N)=O)=O)CC2C)ccc2nc[nH]c2c1F C1(NC(C(C=C)(F)F)=O)CC2CN(C(c3cnc(C(C)C)[nH]3)=O)CC2C1 CCC(CC(=O)N1CC(CN(C(=O)C(C2CCCCC2)O)C)C1)OC C(=O)(C1=CC2(CCOCC2)C1)NCC1CN(C(C(c2cn(C)nc2)O)=O)C1 N1(C(c2c(OCC)scc2)=O)CCC12CN(C(C13COCC1C3(F)F)=O)C2 C(=O)(CC(C=C)CC)N1CCC(C(C(=O)OC)(F)F)(C(=O)OCC)C1 C1(NC(=O)Cc2ccoc2)COC2(CCCN(C(=O)C3=C(Cl)CCCC3)C2)C1 c1(CC)c[nH]cc1C(=O)NCCN(C1CCCCC1)C(C12CC(C)(C1)C2)=O N1(CCC(=O)N(CCCC=C)C2CC2)CCS(=O)(=O)C(CO)C1 c1(CCC(=O)OCC2(C(=O)OC)CC(F)(F)C2)c(C)nc2nc(CN)nn2c1C C1(NC(C2(CC)CCCO2)=O)CN(C(c2cc(Cl)cs2)=O)CC1C(F)F C1(C(C)NC(c2ccc(SC)s2)=O)CCCCN1C(c1cn(C2CC2)nn1)=O O=C(C#CC1CC1)NC1CCCCC1CNC(=O)CCC1CCOC1 c12c(cccc1Br)S2.c1(-c2sc(C)c(C)n2)ccc(C(N)=O)cc1F C1(C(N2CCOC(CNC(=O)CSCC(F)(F)F)C2)=O)(OC)CCC12CCC2 c1(CCC(=O)OC)cnc(N2CCN(C(=O)OC(C)(C)C)CC2)cc1C CC1CN(C(c2cc(N)ccn2)=O)CCC1CNC(=O)CSc1nncn1C1CC1 Cc1cc(N(C)C(c2ccncc2)=O)cc(F)c1.c1(C)nc[nH]c1C CC1Cc2cc(S(=O)(=O)NC(C3CCOCC3)CCOCC)ccc2O1 c1(CNC(CCN(C(C2C(C)OCC2)=O)CCO)=O)cccnc1Cl c1(C(N2CCC(CC(=O)N(CC(C)C)CCC)C2)=O)cccc(Cl)n1 N1(C(c2ccc(C(C)=O)o2)=O)CC2CC(C1)N2C(C1CCCSC1C)=O N1(C(C(Cc2ccc(OC)cc2)C)=O)CCCC(CCNC(=O)C(C)(Cl)Cl)CC1 CCN(OC)C(=O)CNC(C1CCCN1C(=O)C(C)(C)CO)=O C(=O)(CCCCCCNC(=O)COC1CCCOC1)N(c1c(C)noc1C)CC C(=O)(CC(F)(F)C(C)(F)F)NCC(CN(C(CC(c1c(C)noc1C)C)=O)C)O CCC(CC(F)(F)F)C(=O)NC1C2CN(C(c3c(C)nn(C(C)C)c3C)=O)CC12 C(C(C)(O)CC(=O)NC1(CC(N2CC(S(C)(=N)=O)C2)=O)CCC1)OC c1(N2CCC(C(C)C)C2)nc(=NC(C)c2ccc(Cl)s2)[nH]c2c1CCCCCC2 C(=O)(C1=CCOCC1)NCC=CC(C)NC(C1(CC(=O)OC)CC1)=O N1(C(C2CCC(C)N2C(=O)C(C)NC(N)=O)=O)CC2(CNC(=O)N2C)C1 C1(CCCN(C(C2CCN(C(=O)Cc3ccccc3)C2)=O)C2CC2)CCOCC1 c1(C(=O)NC2CC(NC(CC(c3c(C)cccc3)C)=O)C2)ccc(Cl)c(O)c1N c1(C(=O)NCC(N2CCN(C(CC(CC)C)=O)CC2)=O)cc2cnn(C)c2s1 Cc1cc(C(=O)NCC2C3CN(C(=O)OC(C)(C)C)CC23)oc1C C1(C(=O)NC2(C)CC(C(=O)OC)NS2)CCCCC(=O)N1 c1(CCC(N2C(CNC(C3CC3(F)F)=O)CCC2)=O)ccc(C(F)(F)F)cc1 C1(CCCNC(=O)CCc2ccccc2)CN(C(=O)CCn2cnnn2)CCO1 CC1CCCC(C(N2CCSCC2C(=O)N(C)C)C(=O)NC2CCOCC2)C1 C1(CS(C)(=O)=O)(C(=O)NC(CC)(C)CNC(=O)CCCSC)CC(F)(F)C1 N1(C(C(C)(C)CCC#N)=O)CCCC(C2CCN(C(=O)CC3CCSC3)CC2)C1 C1(NC(C2C(C)CCOC2)=O)CN(C(=O)C(F)(F)C(C)(C)O)CC1C1CC1 C1(NC(C(C(C)O)C)=O)CCCN(C(c2cccn(CC(C)C)c2=O)=O)CC1 C1(NC(C2(C(C)C)CC2)=O)C2CCCN(c3ncc(O)cn3)C2C1(C)C c1(OC)cnncc1C(=O)N(C)CC1COCCN1C(c1c[nH]c(=NC)o1)=O c1(N(C)Cc2ccc(C(F)(F)F)nc2)ncnc(N(C)CC2CCNC2)n1 N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CCCN(C(=O)CC2COCCO2)C(C)C1 c1(NC(NOCCC(C)(C)C)=O)cccc(C2CCC(=O)N2)c1 C1(C(=O)NCC2C(CC(=O)NC(C3CCCC3)CC)C2)CC(=O)CS1 c1(OC)c(C(=O)NCC(Cc2ccccc2)NC(=O)C2CC2)csc1C C1(C(N2C(C)CC(CC(=O)N(C)Cc3ccsc3)C2)=O)CCCC(=O)N1C c1(C(=O)NCCCCCN(C(CCc2ncc(C)[nH]2)=O)C(C)C)ccncc1N c1(NCC2N(C(CS(CC)=O)=O)CCCC2C)ncc(Br)cc1[N+](=O)[O-] C1(CCNC(=O)CC2CCCN2C(=O)Cn2cc(Br)cn2)CCCOC1 c1(CC)cc(CC(=O)NC2CC2NC(c2occc2COC)=O)on1 c1(N)ccc([N+](=O)[O-])cc1C(=O)N(C)CCCC=C.c1(O)ccccc1 C1(C(N2CCC(OCC)CC2)=O)CCC2(CCOCC2)CO1.C(=O)(OCC)NCC C1(C(=O)NC2(COCC)CC2)CCN(C(C2CC2(C)CC)=O)C12CCC2 C12(C)CCCN(C1)C(=O)N1CCC(CC1)CN(C)C2=O.C1(C2CC2)(N)CC1 C(=O)(C#CC1CCCO1)NC(C1N(C(c2cc(CCC)c(C)s2)=O)CCC1)C C12(C(=O)NC(c3nc(CC)[nH]n3)C)CC(CO1)N(C(=O)C=Cc1ccsc1)C2 Cc1cc[nH]c1C(N1CCCC1C1(C(=O)NCC(F)F)CC1)=O N1(C(c2c(C)cns2)=O)CCC(NC(c2cc(C(F)F)nn2C)=O)C(CO)CC1 CC1(C)CCCOC1CC(N1CCOCC1CNC(=O)C=Cc1cnc[nH]1)=O N1(C(c2ccns2)=O)CCN(C(=O)Cn2ccnn2)C(c2cccnc2)C1 c1(C(=O)NCC2CCC(NC(C3(CCC=C)CC3)=O)C2)c(C)ccc(F)c1N C1(C)(C(N2CCCC(C(=O)OC)C2)=O)CCCN(c2ncc(Cl)cn2)C1 O=C1CCC2CN(C(=O)NCCC3CCCCC3(F)F)CC2N1 CC(C)(C)C(=O)C(=O)NC1CC(NC(C2(c3cnsc3)CCOC2)=O)C1 c1(C(N2CC(CNC(C(C)SCCCC)=O)OCC2)=O)cc(Cl)ncc1Cl c1(OC)cc(F)c(C(=O)NCCCNC(c2cnn(C)c2C(C)C)=O)c(F)c1F CC(C)(CCl)C(=O)Nc1ccnc(C(=O)Nc2ccc(C(N)=O)s2)c1 Cc1cc(Cl)ccc1C(N1CC(NC(N(C)Cc2ccccc2)=O)C1)=O c1(C(N(CCCCN(C(=O)CCC2(C)CC2)C)C)=O)nnn2c1CSCC2 c1(C(N2CC(O)CCC(NC(c3c(C)scn3)=O)C2)=O)nncc2c1CCCC2 Cc1ccc2scc(C(=O)NC(C)CCN(C(=O)CCCC(C)(F)F)C)c2c1 C(=O)(CCCCCC#N)NC(C(=O)NCCSCC)Cc1ccco1 CC(C)C(C)C(=O)OC1CC(F)(C(c2nnnn2CCOCC2CC2)NN(C)C)C1.CO c1(CC(=O)NCc2cccc(NC(C3(CF)CC3)=O)c2)ccc(F)nc1 C(=O)(CCCCCN=[N+]=[N-])NC(C1CCCOC1)C(=O)NCc1occ(C)c1 N1(C(c2scc(C)c2Cl)=O)CCC(C)C(CNC(C2COC(=O)N2)=O)C1 CC(CCC(=O)NCC1(F)CCC(NC(c2ccc(C(N)=O)o2)=O)C1)N(C)C C1(NC(c2c(CC)ccs2)=O)CC2CCCC(C1)N2C(=O)C(C)=C1CCC1 Cc1cc(C#N)ccc1C(=O)NCC(C)(C)CCNC(c1nnn2c1CCC2)=O c1(CCC2N(C(c3ccc(Cl)c(C)c3N)=O)CCCC2)cccc2ccccc12 c1(C(=O)NCC2COCCN2C(C2CC2F)=O)ccnc2cc(Cl)ccc12 c1(NC(CCNC(=O)CCF)=O)cc(C2CC2)nn1-c1ccccc1 C1(O)(CN(C(CN(C)C)=O)C)CCN(C(c2sccc2-n2ccnn2)=O)C1 c1(OC)ccc(CN(C)C(C)C)cc1OC.N12CCCC1CNC(=O)COCC2 C1(NC(c2cc(N3CCCCC3)ncn2)=O)C2CN(C(=O)COCCF)CC12 c1(OC)ccnc(C(=O)NCC23CCC(CC2)N3C(c2nccc(C)n2)=O)c1O c1(C(N2CCC(SC)CC2C)C(=O)NC)cc(C)ccc1OC(F)(F)F C(CN=c1[nH]cnc2c1CCCC2)(C1CCCCC1)NC(C(CCCOC)C)=O C1(NC(c2nccc(C)n2)=O)CN(C(=O)CC2CC=CC2)CCC1C(F)(F)F C(=O)(C#CC1CCCC1)N1CC(C(N(C)CC2CC(=C)C2)=O)OC(C)C1 c1(C(C)(C(=O)NC2CCC2CNC(c2cc(Cl)no2)=O)OC)ccccc1F N1(c2c(C(CN3C(SCC)CCCC3)=O)cccc2)CCC(C(N)=O)CC1C CC1(C)CC(NC(C2CCOC2(C)C)=O)CN(C(c2cn(C3CC3)cn2)=O)C1 c1(CC)cnn2ccc(C(N3CCC(C)(C(=O)Nc4c(Cl)cnn4C)C3)=O)nc12 C1(C(N2C(C3CCN(C(C=NOC)=O)C3)CCC2)=O)CCC(=O)N(C)C1 CCC(C(=O)N1CC2CC2(CNC(c2cc(CN(C)C)on2)=O)C1)C(C)C c1(OC(C(=O)OC(CCC)(C)C)CC)ccc(F)cc1 c1(C(=O)NC(CN(C(CCSCCC)=O)CC)C)cnn(C)c(=O)c1 N1(C(C2(CC=C)CCOC2)=O)CCC2CN(C(c3cccc(CCO)c3)=O)C2C1 c1(C(=O)NC2CCC(CNC(c3cccc(=O)o3)=O)C2)cncc(O)c1 c1(N(CCC#N)C(CNC(C(C)SC)C)=O)cccc(C)n1 c1(C(=O)NC2C(NC(CCCC=C)=O)CC2)cc(C#N)n(C)n1 C1(NC(C2(SC)CN(C(=O)CCn3ccnc3C)C2)=O)CC(=O)N(C(C)C)C1 Cc1cc(C)c(C)c(C(=O)NC2CN(C(=O)C3=NOC(C)(C)C3)CC2O)c1C N1(C(C2CN(C(C)=O)C2)=O)CCN(C(=O)N(c2ccc(Cl)c(F)c2)CCO)CC1C CCC(C(=O)NCC(O)CNC(=O)C(C#N)=CC1CC1)c1ccco1 CCCC(CNC(c1ncc(F)cc1F)=O)C(=O)Nc1cc(F)ccc1O O=C(O)C#CC(=O)Nc1cccc(CN2CCCC2c2ccccc2)c1 C1(NC(c2c(OC)ccnc2)=O)CCC2CCN(C(=O)CN3CCSCC3)C1C2 c1(OC)c(NC(C2CN(Cc3ccc(F)c(C)c3)CCS2)=O)cc(F)cc1F c1(C2C(NC(C3CC(NC(=O)OC(C)(C)C)C3)=O)CCC2)cc2n(c1)CCOC2 c1(-c2ccc(C)cc2)n[nH]c2c1CN(C(C1CC3CCC1C3)=O)CC2 c1(C(N2CC3C(NC(C(C)(CO)OC)=O)(C3)C2)=O)cccc(Cl)c1F N1(C(c2c(C#C)c[nH]n2)=O)CCC(CO)C(NC(c2cc(C(C)C)n(C)n2)=O)C1 C12(CNC(=O)Nc3scc(-c4ccc(OC)cc4)n3)CCC(CC1F)C2 N1(C(=O)Nc2nc(CN3CCCCC3)cs2)CC2OCOC2C1 N1(C(C(=Cc2cn[nH]c2)C)=O)CC2CCN(C(c3ccc(Cl)c(Cl)c3)=O)CC2C1 N1(C(c2n[nH]c(C)c2C)=O)CC(C(=O)NCCC(C)O)C(C2CC2)C1 c1(C2(C(N(CCN(C(CCNC(C3C(C)=C3)=O)=O)C)C)=O)CC2)cc(C)on1 c1(C(N(CCCNC(=O)Cc2cc[nH]c2)C(C)C)=O)cccc2c1OC(C)C2 C1(CNC(C=CCNC(c2cc(C(C)C)no2)=O)=O)CCCC12CC2 C1(NC(C2CC(C)(C)OCC2)=O)CN(C(=O)C(F)=CC2CC2)CCC1(C)C c12cncc(c1)CNC2.C1(C(N2CCCCC2)=O)CCCN(Cc2ccncc2)C1 CN1C(=O)CCCC1C(=O)NC1CN(C(=O)C=CSc2ccccc2)CCC1F N1(C(C2CN(CC)C(=O)N2)=O)CC2CC1CN2C(=O)C(C)(Cl)Cl N12CC(CC(C)(C)C1)NC2=O.C(CCN(C)C)(C(C)(C)C)OCC C=CC1OCCCC1C(=O)NCC1CC1NC(c1cc(CC)oc1C)=O N1(C(CCC#C)=O)CCN(C(CNC(=O)CCC(=O)OCCC)C(F)F)CC1 CN1CCCN(C(=O)CC(C2CC2)NC(C2CCC(=O)N(C)C2)=O)CCC1 Cc1cn2ccnc(C(=O)NC3CC(CNC(=O)CCCC#N)C3)c2n1 Cc1ncc(C(N2CCCC2C2(NC(C3CC(=C4CCC4)C3)=O)CC2)=O)cn1 N1(C(Cc2cc(COC)on2)=O)CC(C)C(C)(CNC(c2c(C)ccnc2O)=O)C1 C1(NC(=O)Cc2n[nH]cc2Br)(CNC(c2ccccc2)=O)CCCCCC1 Cc1cccc(CC(=O)NC2CCN(C(c3cn(C(C)C)cn3)=O)C2)c1 N1(C(c2nccc(OC)c2)=O)CCC(NC(=O)CC2CCC(=O)N2C)C1(C)C c1(NCC(CNc2ncc(C(=O)OC)c(C)c2)C)cc(F)cc2ccoc12 C1(F)(C(N2CC(SC)C(NC(c3cccc[n+]3[O-])=O)C2)=O)CCCN(C)C1 Cc1c(C(N2CC(N(C)Cc3c(Cl)cccc3I)C2)=O)nc2ccccn12 c1(CNC(COC2CCN(C(c3c[nH]c(=NC)s3)=O)C2)=O)ccc(C)c(F)c1 C1(C(=O)NCCC(C)N(C(c2cnc(SC)s2)=O)C)CCC2(COC2)OC1 C1(CC(=O)NC2CN(C(=O)CC3(O)CC3)C3(CCC3)C2)COc2ccccc2O1 c1(NC2(CNC(CC(CC)c3ccccc3)=O)CC2)ncnn2cccc12 CN1CCC(C)(C(N2CC3(CCN3C(=O)CCc3ccc(F)c(F)c3)C2)=O)C1=O c1(C(N2CC(O)(C(C)(C)CNC(=O)Cc3cnco3)C2)=O)cccc2sncc12 n1(CC(=O)N(C(C(=O)NC(c2nc(C)on2)C)(C)C2CC2)C)nc(C)nc1C CC(Cc1ccccc1)C(=O)NCCNC(=O)CC12CC(C1)C2 c1(CC)cc(C(=O)NCC(CNC(=O)Cc2scnc2C)OC)sc1C Cn1cnc(C(=O)NCC2CC(O)(CNC(c3cc4ccsc4s3)=O)C2)cc1=O c1(CC(O)COC(c2nc[nH]c2Nc2ccccc2)=O)ccccc1Br C1(C(=O)NC(CC=C)CNC(=O)CCCn2ccnc2C)(OC)CCOCC1 c1(C(=O)NC(C2CCCN(C(=O)COCCF)C2)C)cnc2ncc(Cl)cn12 N1(C(C(=Cc2ncn(C)c2)F)=O)CC2(CCN(C(C3CCCOC3C)=O)C2)C1 CC1COCCC1N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC3CCC3)cc2s1 Cc1ccn(C(C)C)c1.c12cnn(c1)C1(C(=O)NC3(c4ccccc4)CC3)C2C1 CCC(C)CCCC(=O)NCC(C)(C)CN(C(=O)C(O)C1CCC1)C C(=O)(C1=C(C#N)CCC1)N1CCCC(C)(NC(c2sc(C)c(O)n2)=O)C1 N1(C(c2c(C)c[nH]n2)=O)CCN(C(c2ncc(Cl)cc2F)=O)CC1C(C)C C1(NC(CN(C(c2ccno2)=O)CC)=O)COCC1NC(c1ccccn1)=O.CC N1(C(C2C(C)C2C)=O)CC(NC(=O)CCCCNC(N)=O)C(O)C1 Cc1cc(CNC(C2(CNC(C3CC(F)(CF)C3)=O)CC3(CC3)C2)=O)oc1C N1(C(c2c(C(C)(C)C)con2)C2CC2)CCC(c2ccccc2)C(C)(C)C1 C(=O)(C(O)CN1CCC1)NCCC(C)N(C(CN(C(C)C)C)=O)C CC1C(N(C)C)CCN1C(=O)C1CC1.C1(=O)C(C)N1 C#Cc1cc(C(N2CCCCC2CCN(C(=O)C(C=C)OC)C)=O)ccc1C c1(C(=O)NCCCN(C(C(CSC)C)=O)CCO)ccn(C(C)C)c1C Cc1ccc(S(=O)(=O)N(C(C)(C)C(F)(F)F)C2CC2)c(Br)c1 C=CCC(CC(C)C)C(=O)NCCCC1CCCN1C(c1ccncc1F)=O C1(C)(CNC(C(N2CCC(C)C2)=O)=O)CCCN(Cc2nnc(C(F)F)s2)C1 c1(NC)ccccc1C(=O)NC(CNC(=O)CC(c1ccc(N)cc1)C)C(C)C c1(C(N2CCN(Cc3c(OC)ccs3)C3C2C3)=O)ccc2nc(C)sc2c1 C1(NC(C2C(CNC(Cc3nc(C)sc3)=O)OCC2)=O)CNC(=O)C1(C)C C1(CNC(c2c(C)nns2)=O)(NC(c2ccsc2)=O)CC2CCC1CC2 c1(CN2CC(CC(=O)NC3CC4(CC4)C3)C2)cc2ccccc2cn1 N1(C(C2(C)CCN(C(CC(=O)NC)=O)C2)=O)CC2CCCC(C2)C1 N1(C(COCCCC)=O)CC(NC(=O)CC2C=CS(=O)(=O)C2)C(S(C)(=O)=O)C1 N1(C(C(C)OCCC(C)C)=O)CCN(C(=O)CN2CC3CC3C2)C(C(C)C)C1 C=CCC(C(=O)NCC1CCCCN(C(c2cncc(N)c2)=O)CC1)C(C)C C1(C2(O)CCN(C(=O)C=CC(C)(C)OC)CC2)(NC(C(CC=C)NC(C)=O)=O)CC1 c1(CCC(=O)NCC2CCN(C(=O)CC3CCOC3)C2)ccc(C(F)F)cc1 c1(OC)cc(C(=O)NC2CCCC2C(=O)Nc2cccc(F)n2)ccc1C#N S(=O)(=O)(c1cnccc1N1CCOC(C)(C)CC1)N(CCC(F)(F)F)CC CCC(C)C(C(=O)N(C)Cc1occc1C)N(C(=O)C(C(C)OC)N(C)C)C N1(C(c2cc(CNC(C(C)n3cccc3)=O)[nH]n2)=O)CC2CCCC(O)C2C1 Cc1cc(C)c(C)c(C(N2CC=CC(NC(=O)CC3CCCO3)C2)=O)c1C N1(C(C2(CC#C)CCN(C(c3scnc3C)=O)C2)=O)CCCOC(C)(C)C1 C12(C(=O)NCc3scc(CNC(C4CCC(C)O4)=O)n3)CCC(CC1)CO2 Cc1cccc(C)c1CC(=O)NC(CO)C(C)NC(C1(F)CC2(CCC2)C1)=O C12(CNC(C3C(C)C3C3CC3)=O)CCC(NC(=O)COc3cnn(C)c3)(CC1)CO2 C1(NC(=O)CC2CCCN2Cc2cccc(Cl)c2)CC2(CCC2)C1 Cc1cc(C)c(C(=O)NCCC23CCC2CN(C(C2(N(C)C)CC2)=O)C3)cc1N C1(C)(C(=O)NCC2(COC)CN(C(C(CC)OC)=O)C2)CCN(C(C)(C)C)C1 N1(C(=O)C=Cc2cccc(O)c2)CC(NC(C2CC(F)C2)=O)CC12CCOC2 N1(C(C(CC)O)=O)CCC(O)(CNC(=O)C(C2CCCCC2)OC)CC1 N1(C(c2cc(CC)n(CCO)n2)=O)CCC2CN(C(C3CCC3)=O)CC2CC1 N1(C(C(C(C)O)C)=O)CCC2(COC(CNC(c3ccc(CCF)cc3)=O)C2)C1 c1(C(N(CCC)CCNC(=O)CSCCN(C)C)=O)ccc(C(F)(F)F)o1 n1(C(C)C(=O)NCC2CCCCN2C(=O)Cn2ncnn2)cnc2ccccc12 c1(C(N2CC(O)(C(C)NC(C3C(CCOC)C3)=O)C2)=O)cc2ccc(Cl)cc2s1 CC1(C)COC(C(=O)NCC(C2CCCC2)NC(=O)C=Cc2ccccc2)C1 c1(NC(C2C(Nc3c(C)cncn3)C2)=O)ccc(-c2ccccc2)nc1Br C12(NC(C3CC(CN(C)C)C3)=O)CC1CCN2C(C1COCC1C(N)=O)=O N1(C(CC2N(C)CCOC2)=O)CCN(C(c2cc3c(ccn3C)[nH]2)=O)CC12CCC2 c1(CN2C(C(=O)Nc3n(COC)ncc3)CCC2)nccc(Br)n1 Cc1cc(C(=O)NC2CC3(C2)CN(C(C2(C)CCCS2(=O)=O)=O)C3)nc(C)n1 N1(C(COCC=C)=O)CCCCC(CNC(C2(CCOC)CCC2)=O)C1 C1(CNC(COCC)=O)CCCN(C(c2n[nH]cc2F)=O)C1 N1(C(=O)CSC2CCCCO2)CCCCC1C1CCCN1C(C12CC3CC1C2C3)=O C12(C(=O)NCCNC(CCCNC(=O)OC(C)(C)C)=O)CCCCC1C2(F)F Cc1csc2ncc(C(=O)NCC3CC(C)N(C(=O)CCCCC(N)=O)C3)n12 C1(C(=O)NCC(=C)CCNC(C2CCCN2S(C)(=O)=O)=O)CC2CC(OC)C2C1 C(=O)(CC1CCOc2ccccc21)NC1C(NC(CCSCCC)=O)CCC1 CCC(CC(=O)NC1CCC1CNC(C1(c2ccccc2C)CC1)=O)C(C)(C)C c1(C(=O)NC(C2CCN(C(c3cn(C)cn3)=O)C2)C)cccc2cnsc12 C(N=c1[nH]c(N2CCn3c(CC)nnc3C2)nc2c1CCC2)C1(CCC)CCC1 N1(C(C(C)OCC2CC2)=O)CC(NC(=O)CC2CCC(C(F)(F)F)O2)(OC)C1 C1(NC(c2c[nH]nc2C2CC2)=O)CCN(C(c2cnco2)=O)C12CC2 c1(C(N2CC(NC(c3coc(Br)c3)=O)C2)=O)cc(=O)c2cc(Cl)ccc2o1 CC1=C(C)CN(C(=O)CCN(C(=O)CN2CCCC2=O)CCO)CC1 CC(CC(N)=O)C(=O)NC1CCC(NC(=O)CCCn2cncn2)CC1 c1(C(C)=O)cnc(N2CC(NC(c3cc(O)ncn3)=O)CCC2C)c(C)c1 C12(CNC(NCC3(COC)CCCC3)=NCCF)CCCC(C1)C(=O)N2 c1(NCCC(C)NC(C2(OC)CCCC2)=O)nc(Cl)nc2c1cnn2C c1(C(N(C2CCN(C(C3CN(S(C)(=O)=O)C3)=O)C2)CC)=O)ccc(OC)cc1 c1(C(=O)NC(CC=C)CNC(=O)CC2CSCCS2)ccc(C#N)c(C)n1 c1(NC(N2C(C(=O)NCC(C(=O)OC)O)CC2)=O)n[nH]c(C)c1F.C(C)(C)(C)O Cn1cnc2cc(C(=O)NCC(CNC(C3(F)CCC3)=O)CO)cnc12 Cc1nn(CC(O)CNC2CCCN(C(=O)OC(C)(C)C)C2)cc1I C1(CCNC(C=CCCC(C)C)=O)CC2CCC(C1)N2C(c1csc(F)c1)=O C1(CNC(C(C=C)O)=O)CN(C(=O)CC2(CO)CCCCC2)CC(C)(C)O1 N1(C(CNC(c2ccn(C)c2)=O)=O)CCN(C(c2cn(C(F)F)cn2)=O)CC1 c1(CN2C(C(N3CCC(COC)CC3)=O)C=CC2)c[nH]c2cc(F)c(F)cc12 C(CC(C)C)(C(=O)NCC1CCN1C(=O)C(c1ccc(Cl)cc1)=O)NC(C)=O C1(C(=O)OCc2ccn(CC)n2)C(NC(C)=O)C2CCCCC12 C1(C(=O)NC2(C)CN(C(=O)CCCc3ccncc3)C2)CC12CCCOC2 Cn1cc(C(F)=CC(=O)NCC2CCCCN2C(C2OCCC2(C)C)=O)cn1 C1(CNC(C)(C)C)CN(C(c2cccc(C(=O)OC)c2F)=O)C(C(=O)O)CC1O C1(CNC(C2(C=C)CCC2)=O)CCCCN(C(=O)CN2CCC(C)(O)C2)C1 c1(C(=O)N(C2CCNC2)C2CC2)c(F)ccc2[nH]ccc12 CC1(C(=O)NCC2CCCN2C(=O)CSC(F)(F)F)CC=CCC1 C(=O)(C1CCCc2ncccc21)NC(CC)CNC(=O)C=C(C)c1cccs1 N1(C(C2N(C)CC(C)(C)C2)=O)CC(C)(C)CCC1CNC(C1(F)CCCCC1)=O c1(C(=O)NCC(N(C(C(C)CC(F)F)=O)C)C2CC2)[nH]cc2c(=O)n(C)ccc12 C1(NC(c2ccc(C(C)C)o2)=O)CN(C(=O)CC23CC(C2)C3)C2(CCOCC2)C1 c1(C(N(C)CC2N(C(c3c(OC)cccn3)=O)CCC2)=O)nn(C)c(C)c1Cl C(CCN=C(NCCC(=O)N(C)C)N1CCC(C)(c2ccccc2F)C1)CSC N1(CC(C)O)C(=O)NC(Cc2ccc(-c3cccc(-n4cccn4)c3)cc2)C1=O CCC(C)CCCC(=O)NCC(CC(=O)N(C1CC1(C)C)C)OC C12(C(=O)NCc3oc(C)c(C(=O)NCCOCC4CCC4)n3)CCC(F)(CC1)C2 c1(SCC#C)cccc(C(N2CCC(NC(=O)CCc3cnn(C)n3)C2C)=O)c1 O=C(C(F)C1=CCCCC1)NC1(CF)CCN(C(=O)CN2CS(=O)(=O)C2)C1 Cc1nc(NC(CNC(=O)C=Cc2cnccc2C)C(C)C(C)C)cc(C#N)n1 c1(C(=O)OC(C(CC)C2CCOCC2)=O)cc(C)ncn1 Cc1ccc(OC(C2CCOC2)CNC(=O)CNC(C)(C)C)cc1 Cc1nc(C(N2CCC(N(C)C(C3CC(N(C)C)C3)=O)C2)=O)c2ccnc-2[nH]1 N1(C(c2nc(C(C)C)oc2)=O)CC2C(CN(C(=O)CCNC(=O)C=CCl)C)C2C1 Cc1nc(S)sc1CC(=O)NC1CCCN(C(=O)CCc2nc(C)c(C)o2)C1 Cc1nn(C)c(NC(C2CCN(Cc3cnc(C(F)(F)F)s3)CC2)=O)c1C=O C1(C(=O)NCCN(C(C)C)CCN2CCCC2C(=O)N(C)C)CCC(F)(F)CC1 c1(CNC(c2ccc(OC3CCC3)cc2F)=O)ccc(Cl)cc1F C1(NC(CCc2c(C)nn(C)c2)=O)CC2CCC1N2C(=O)CCCC(=O)C1CC1 C(=O)(C(O)C(C(C)C)OC)NC1CC(CNC(c2cc(OC)cc(OC)c2)=O)C1 N1(CC)CC(NC(C2CC3CC3N2C(=O)CCc2nc(O)n[nH]2)=O)CC1=O c1(C(N2CCCC(NC(C(COC)O)=O)CC2)=O)cccc(S(=O)(=O)N(C)C)c1 c1(CC)cc(Cl)ccc1Cn1cc(C2(C(N3CCCC(O)CC3)=O)CCC2)nn1 CC(CCCNC(c1ncc(C(F)(F)F)s1)=O)NC(c1ccsn1)=O c1(C(=O)NCC=CCNC(C2(C)CCCNC2=O)=O)cccc2ccncc12 CC(CC#N)C(=O)NCCC(=O)NCC1CCCCN1C CC(C)C1=NOC(C)(C(=O)NCC2CN(C(=O)Cc3sc(O)nc3O)CCO2)C1 N1(Cc2ncc(C(=O)OC)o2)CCCCC(CO)C1.c12ccc(c(O)c1)oc2=O N1(C(C(CC)C(C)O)=O)CCCC(C)(C)C1CNC(=O)Cc1ccc(OC)cn1 C1(NC(C(c2cnn(C)c2)C)=O)CC1C1CCCN(C(c2cnnn2C)=O)C1 C(CC(C(=O)NCc1ccns1)NC(c1ccn(CC)n1)=O)OCC C1(C(=O)NCC(C)(C)C(N)=O)C2CC3C1C3C2N c1(CC(=O)NC2C=CC(C(=O)NCC3CCC34CCC4)C2)ccc2c(c1)OCO2 c1(NS(CC)(=O)=O)ccc(C(=O)NCCCNC(=O)CCC(C)SC)cn1 C1(C(N2C(CCNC(C=CCN(CC#C)C)=O)CCC2)=O)CC(=O)NC(C)C1 C(=O)(C(C)CC(C)(F)F)N1CC(NC(Cc2nccc(CC)n2)=O)CC12CCC2 c1(C(=O)NCCN(C(c2scnc2Cl)=O)C2CC2)cncc2n[nH]cc12 c1(C(=O)NCC2CCN(C(C(CC)C(C)O)=O)C2(C)C)coc(S(C)(=O)=O)c1 N1(C(C(n2c(C)cc(C)n2)C)=O)CCCN(CCNC(=O)C(C)C2CC2)CC1 C12(NC(COCC(C)(C)C)=O)CCCN(C(c3cnc4n3CCC4)=O)CC1C2 c1(SC)ccc(Cl)cc1F.c1(C(CC(C#N)NC)C(=O)N)c(Br)cnn1C c1(CN2CC(CN)OCC2)nc2c(s1)CCCC2 C1(COC)(CNC(C2CCN(C3COC3)C2)=O)CN(C(c2ns[nH]c2=O)=O)C1 C(=O)(C#CC1CCOCC1)NC1CC(C(=O)NC2CC(C)(C)OC2)CC1O Cc1cc(CC(=O)NCC(=O)N(C)C)cs1.C12(CC1)C(=O)N2 N1(C(CCOCC(C)C)=O)CC(n2cc(C(=O)OCC(F)(F)F)nn2)C(C)C1 C(N=c1[nH]c(=NCC(C)S(C)(=O)=O)[nH]c2cc(COC)ccc12)C1(COC)CC1 N1(C(c2ccc(CCCC)cc2)=O)CC2CN(C(c3cc(C)nnc3O)=O)CC2C1 N1(C=O)CC2CC1CC2CN1CCSCC1.c1(C)cc(N2CCOCC2)ccn1 Cc1c(-c2cn(CC(C)(C)CNC(=O)C(C)OC(C)(C)C)nn2)cccc1Br O=S(=O)(c1ccc(NCC(CO)CC(F)(F)F)c(Br)c1)NCCC1CCOC1 Cc1c(CCC(N2CCOC(CN(C(=O)Cc3ccsc3)C)C2)=O)cnn1C c1(CC(N2C(C(=O)NCC(C=C)OC)CSC2)=O)c(C)nc2ncnn2c1C c1(NC(C2COCCN2Cc2cncc(Br)c2)=O)cc2ccccc2c(Cl)n1 Cc1cncc(CC(=O)NCC2(C(C)(C)C)CCN(C(=O)C=CS(C)=O)C2)n1 C(=O)(CCN(OC)C(=O)c1c(C)ncnc1C)N.C1(C(=O)OC)CN(C(C)=O)C1 CC12COCCN(C1)C2.C1(OCC(=O)NCC2CCCO2)CCCCC1 N1(C(CCCC)=O)CC2(CCOCC2)CC1CNC(C1CCC(C)(C)O1)=O N1(CC(=O)N(C(CNC(C)=O)C(F)(F)F)CC)CCC(OC)C1(C)C c1(C(=O)NCC(C)N(C(c2ccc(CC)s2)=O)C)c(OC)cnc2ccccc12 N1(C(C=NOC)=O)CC2CN(C(C3CCN(C(=O)CC(C)C)CC3)=O)CC2C1 CCCCCC(C)CC(=O)N1CCC(C)(C(=O)N(C)CC2CCOC2)CC1 CCC(O)CN(C(=O)CC1(N(C(=O)CCOCC(C)C)C)CC1)C1CC1 C(=O)(C1CCCc2ncnn21)Nc1nc(C)nc(N2CCC3(C2)OCCCO3)c1 C1(C(C(=O)OC)N(C(=O)CCN2CCCC2)CC2CC2)CCOCC1 C#Cc1cccc(C(=O)NC2CC(C(=O)NC3CCC(CC)CC3)C23CCC3)c1 c1(C(N2CC(CC(C)NC(C(n3c(C)ccn3)C)=O)C2)=O)ncc(N)cc1Cl C1(NC(C(CCC)N(C)C)=O)CC2CC(C1)N(C(c1nc[nH]c3ncnc1-3)=O)C2 C(=O)(C(C)(C)C(C)C)N(C1CCN(C(=O)CCCF)CC1)CCCC N1(CCN(C(CC2(CC=C)CCCC2)=O)C)CCN(C(C2(C)CC2(F)Cl)=O)CC1 C=CCC(C)(C)C(=O)N1CC2(CCC2NC(c2cc(-c3ccoc3)[nH]n2)=O)C1 C(CO)(C(=O)NCc1nc(C(=O)NCC2CCCN2C(C)=O)co1)OC CC(O)CCCCCC(=O)N1CC(NC(=O)CCNS(C)(=O)=O)C1 C1(C(=O)NCCSCC(=O)OC)CCN(C(=O)C2CC3CC2CC3O)O1 N1(C(CC(C)OC)=O)CCCC12CCN(C(=O)C(c1ccccc1Cl)(F)F)C2 C1(c2cn(C)nc2)CCC(N=c2[nH]c(=N)[nH]c(=NCc3csnn3)[nH]2)C1 CN1CCc2c(C(N3CC4CC(C(N)=O)C3C4)=O)cccc21.C1(C(=O)N)(CF)CC1 C1(C(C)NC(C2CC(C#N)C2)=O)CCCN(C(c2cccnc2Cl)=O)C1 N1(C(c2c(C)c(Br)ccn2)=O)CC(NC(=O)CCC2CCOC2)C(C2CC2)C1 C#CC1(C(=O)NC(c2ccc(C)nc2)C)CCN(C(c2ccnc(OC)c2)=O)C1 c1(C(=O)NCC(CNC(c2n(CC)nnc2)=O)O)cc(C2CC2)ncn1 Cc1ncc(Br)c(C(=O)NCC2(NC(C3CCCC3C(F)(F)F)=O)CC2)n1 C(=O)(CCC(=O)N1CC(NC(=O)Cc2c[nH]nc2C(F)(F)F)C1)N(CC)CC N(C1CCCc2c(Br)cccc21)C(c1c2cnn(C)c2ncn1)=O C1(C(=O)NC(CN(C)C)CO)CN(C(C2CC2Cl)=O)CCN1C C1(CNC(=O)Cc2cncnc2)CCC(C(=O)NCC2(CCCCO)CC2)O1 c1(OCC)ccc(Cl)c(CC(=O)NCCC(C)N(C(=O)CN2CSCC2=O)C)c1 N1(C(CN(CCS(C)(=O)=O)C)=O)CC(C(=O)N(C)CCO)C(C)(C)C1 c1(C(=O)N(CC2(CCOC)CC2)CCl)cc2ccccc2[nH]1.c1(C)c(F)cccc1F C12(C(N3CCCC(N(C)C(C4(NC(N)=O)CC4)=O)C3)=O)CCOC1CC(=O)NC2 C12(C(=O)NC3(C=C)CC3)CCC(CC1)N(C(c1nn(C)cc1Cl)=O)C2 CCC(CC(F)F)C(=O)NC1CC2(C1)CC(NC(=O)CN1CCCCC1)C2 C(=O)(C(C)(C)C1=CCSCC1)N(CC(C)NC(c1c(C(=O)OC)n(C)nc1)=O)C c1(C(=O)NC(CC(C)NC(C23CCC(CC2)C3)=O)C)ccccc1NS(C)(=O)=O N1(C(C2OCCN(C(=O)CC3(O)CCCOC3)C2)=O)CCCC(F)(F)CC1 N1(C(C=CC(CC)C)=O)CCC2C(NC(=O)Cn3nnnc3C)CC12 N1(C(c2n(C)ccn2)=O)CC2CCC(NC(=O)C(C)(O)c3ccccn3)CC2C1 c1(OC)cc(C(N2CCCCC(NC(c3sccc3Cl)=O)C2)=O)c(Cl)cn1 C(=O)(CC1=NN(c2ccccc2)C(=O)C1)N1CC(NC(C2CC3(COC3)C2)=O)C1 c1(C(N(CCC(C)NC(C2CN(C(=O)NC)C2)=O)C)=O)ccnc(O)c1 c1(-c2cn(C(C(=O)NCC3CN(C(C)C)CC3O)C)nn2)ccc(C#N)cc1 c1(C(N2CC(N(C(C(C)CS(C)=O)=O)C)C2)=O)cc2cccc(Br)n2c1 C(C(=O)NCCCN(CCCCNC(c1cn(C)nc1O)=O)C)(C(C)(C)C)OC N1(CC(=O)N(CC)CC)CCC(NC(c2ccc(CC3CC3)s2)=O)CC1C C1(NC(c2cnc(OCC)s2)=O)CCN(C(=O)CCCc2sccc2C)CC1O N1(C(CCc2onc(C)n2)=O)CCCC(C(=O)N(C2CCOCC2)CC(C)C)C1 N1(C(C=C(C)C)=O)CC2(CCNC(c3cccc(O)n3)=O)CCC1CC2 C1(C(N2C3CC(NC(C(CCC)C)=O)(C3)C2)=O)CN2CCCN1CC2 c1(COC)nc(OC)cc(N2CC(NC(C3(C)CC(C)=NO3)=O)C(C)(C)C2)n1 c1(C(N2C(COC)CCC2)=O)cc(C)cnc1NC(C1CN(c2ccccc2)C1)=O c1(C(=O)NCCOCCN(C)C(c2ccc(Cl)cn2)=O)c[nH]cc(Br)c1=N N1(C(c2n(CC)ccn2)=O)CC2(CCN(C(C3CSC(C)=N3)=O)CC2)C1C(C)C S(=O)(=O)(c1cccc(F)c1)NCC(N1CC(O)(CNC(CCCOC)=O)C1)=O C1(NC(=O)Cn2cc(Cl)cn2)CC2CN(C(=O)CC3CSC3)CC2C1 c1(C(N2CC3(CCN3C(c3cc(O)cc(Cl)c3)=O)C2)=O)c(F)ccc(Cl)c1F N1(C(CC(C)(C)SC)=O)CC(CNC(C2CC(F)(F)CS2)=O)CC1(C)C Cc1ccc2c(C(N3CCCC(NC(=O)C(C)(F)C(C)(C)F)C3C)=O)coc2c1 C1(C(N2CC(CNC(C3CC(C)(C(C)C)C3)=O)(OC)C2)=O)(OC)CCSC1 C(C)(C(=O)NC(C(=O)N(C)CCF)c1ccoc1)OCC c1(C(=O)NC2CN(C(c3c(CC)con3)=O)CC2C)noc2ncccc12 c1(N2CC=CC(NC(c3cnc(CCC)s3)=O)C2)ncn(C)c(=O)c1Br C(=O)(C(C)(O)CNC(=O)CC(C1CC1)NC(c1cc(Cn2ccnc2)on1)=O)OC CCCCC(C(=O)NC(C)(C)CCCC(=O)NC(c1ccccn1)CO)C(C)C CCCC(CC(C)C)C(=O)NC(CCF)C(=O)NCc1cc2n(n1)CCC2 C1(c2nnc(C)o2)CN(C(=O)CC2COC(CN)C2)CCO1 C1(COC)(NC(=O)C#CC(C)C)CCN(C(c2ccc(CC(C)C)cc2)=O)C1 C1(CNC(CCc2cc(C)on2)=O)CN(C(c2ccc(O)nn2)=O)C2(CCC2)C1 C1(NC(C(c2ccccc2Cl)C)=O)CCCC(N=c2[nH]c(Cl)nc3c2CCC3)C1 N1(C(c2ccc(Oc3c(C(N)=O)cccc3)cc2)=O)CCOC2CCNCC12 C(=O)(C1=COCCO1)NC1CCCN(C(Cn2c(CCC)ncc2)=O)C1 N(C(=NCCCN1CC=CC1)NC1CCOC(C(=O)OC(C)(C)C)C1)C(CC)C Cc1cnc(C(N2CCCN(C3CC3)CC2)=O)cc1Cl.C(=O)(C1=CCCSC1)NC c1(OC)cc(C2OCCC2C(=O)NCC(C)CN(C(=O)C(F)OC)C)ccn1 c1(C(=O)NCCCCC(C)NC(C(CC)O)=O)cc(F)ccc1N Cc1c(Br)c(C(N2CC(C3(NC(c4cnc(S)nc4)=O)CC3)C2)=O)nn1C c1(C(=O)NCC2CC(O)CN2C(c2cccnn2)=O)c[nH]c2ccc(F)cc12 N1(c2n(CC=C)c(C(c3ccccc3)(C)O)nn2)CC(CC(=O)OC)OC(C)C1 c1(NC(c2c(C)cco2)C)ncnc(N2CC(CSc3cccc[n+]3[O-])C2)c1C N1(CC(=O)NCCC2CC(NC(C(c3ccccc3)C)=O)C2)CCCC1CO CN1C(=O)CSC1=CC(=O)NC1CC2CCC(C1)N2C(c1cnc(O)c(Cl)c1)=O C12(CNC(c3ccc(-c4cn(C)nc4)o3)=O)CC(CO1)N(C(=O)C1=CCC1)C2 C(=O)(C(C(C)C)N(C)C(=O)OC(C)(C)C)NCCCn1c(C)nnc1 c1(C(C)(C)C)cc(OCC(=O)NC2CC2(C)Br)ncn1 Cc1cc(O)nc(C)c1C(=O)NCCCCCCNC(=O)CC1CCC1C(=O)O c1(C(=O)NCC2C(C)CN(C(=O)CCc3nncs3)C2)ccc(F)cc1O c1(C(N)=O)c(C2CCN(Cc3ccc(-c4cccs4)o3)CC2)cnn1C c1(C(N2C(CNC(c3cccc(Cl)c3)=O)CC(OC)C2)=O)cccc(S(C)=O)c1 C1(CN(C(C2CCC(C(C)C)C2)=O)CC)CCCN(C(c2cc(Cl)cnn2)=O)C1 C#Cc1ccc(CCC(N2CCCC(NC(c3cnc(O)n3C)=O)C2C)=O)cc1 C(N1CCN(C(=O)Cc2ccc(F)cc2)CC1)n1c(C)cc(C)n1 S(=O)(=O)(c1ccc(N2CCc3c(Cl)cccc3C2)nc1)NC1C(C)(C)SC1 C1(NC(c2ccc(C(C)C)s2)=O)CC12CC(NC(=O)C(O)Cc1cnn(C)c1)C2 C(=O)(CC(F)(F)C(F)F)N1CC(C)CC(NC(CC(CC)O)=O)C1 CC1CC(CNC(c2coc(C(F)(F)F)c2)=O)CN1C(=O)CCN1CCOC1=O C(=O)(CC(F)(F)F)N(NC(C(=O)NCCNC(C1(C)CCCO1)=O)C)SC(C)(C)C C1(CC(N2CC(C)OCCC2)=O)N(C(=O)CCC2CCC2)CCC1(C)C N1(C(C(C(CC)C)=O)=O)CC2CCN(C(=O)CC3(COC)CC3)C2C1 C(=O)(C#CC1CCCOC1)N(CCNC(C)=O)C1CC1.C12(CCCC1)C(=O)N2 c1(C(N2CCCC(NC(C(C)S(C)(=O)=O)=O)C2)=O)ncn2c1CCCC2 C1(CNC(CC2CCC(OC)CC2)=O)C(C)CCCN1C(C1CC12CC2)=O C1(C(=O)NCC23N(C(CCCC#N)=O)C(CC2)CC3)CCc2ncnn2C1 C1(NC(C(CC=C)C)=O)CCC2(CCN(C(=O)CN3CCCCC3=O)CC2)C1 C1(C(=O)NC2C(OC)CN(C(c3[nH]nc(OC)c3Cl)=O)C2)CCC2CC2CC1 C1(CN(C(=O)C=C2CCSCC2)CC)CCCN(C(=O)C(C)NC=O)C1 c1(NC(C(C2CCN(c3ncc(C)cn3)CC2)C)=O)ccc2ncsc2c1 C1(NC(C=CC(CC)C)=O)CCN(C(=O)CN(C)C2CC2)CC1CO C1(NC(CN(C)C(C2(F)CCOCC2)=O)=O)CCCC2(CCC2)C1 C1(NC(C(C)=C2CC2)=O)CC2(CCN(C(=O)CC3CCCCC3(C)C)C2)C1 C(=O)(CCC(C)(C)C#N)NCC1CCCC(NC(CN(CCOC)C)=O)C1 C1(C2CCCCC2)(NC(C2CCCC(NC(CCC#C)=O)C2)=O)CC1 Cc1cc(C(N2CCC3CCC23CNC(c2cc(Cl)ccc2F)=O)=O)ncc1N CC1CN(C(c2ncccc2C(F)F)=O)CC(C)N(C(=O)CS(N)(=O)=O)C1 C1(C(=O)N(CC(CC)C)CC)CN(C(=O)C(=O)NCc2ccccc2)CC1CO c1(C(=O)NC(C(=O)OC)Cc2c[nH]c3ccccc23)n[nH]c2ccc(O)cc12 c1(-n2c(Cc3cc(OC)c(C)nc3)nc(-c3cscn3)n2)ccc2ccccc2n1 c1(-n2ccc(NC(C3(C)CCOC3)=O)n2)cccc(C(C2CC2)NN2CCCC2)c1 C1(CNC(CN(CCC#C)C)=O)CC2(C1)CN(C(c1ncc(C)cc1F)=O)C2 c1(C(=O)NCC2CCCN(C(c3c(C)cno3)=O)C2)[nH]c(C)c(S(N)(=O)=O)c1C CCC(CN(C)C)CC(=O)N1CCC(C)(CNC(C2CC(F)(CO)C2)=O)CC1 c1(C(N2CC3CC(C2)N3C(=O)C(O)c2ccsc2)=O)cnn2c1OCC2 c1(C(N2CCCC(NC(C3N(C(C)=O)CC3)=O)C2C)=O)cc2c(nn1)CCCC2 C1(C(=O)NCCCCCCNC(CCCOC)=O)CCOC(=O)CC1 C(=O)(CC(C)(C(F)F)N(C)C)NC1(CO)CCN(C(c2c(C)cc(C)nc2)=O)C1 Cc1coc2ccc(C(N3CCC4CCN(C(=O)Cc5ccoc5)CC34)=O)cc12 C(=O)(C(C#N)(CC)CC)N(C)CC1OCCN(C(CN(C2CC2)CC)=O)C1 C1(NC(C2CCN(C(CCC3CC(OC)C3)=O)CC2)=O)CN(C)CC1(F)F Cc1cccc(C(=O)NC(C)C(C)C(=O)N(C)Cc2ccncc2F)c1O C1(CNC(c2nc(C)sc2C)=O)CN(C(c2scnc2C(C)C)=O)C2(CCC2)C1 c12ccnc(c1)NC2=O.Cc1nnsc1C(=O)COC(=O)CC(C1CC1)N(C)C N1(C(C2C3CN(C(c4c(OC)nn(C)c4)=O)CC32)=O)C2CCC1CN(C)C2 c1(NC(=O)C(=O)NC2CC23CCc2ccccc23)cccc2c1CCOC2 c1(C(C(N2CC(CNC(CCCC=C)=O)C(O)C2)=O)N(C)C)ccc(Cl)c(F)c1 C1(NC(=O)C2CC2)CN(C(c2ccn(C3CC3)n2)=O)CC2(CCOCC2)C1 C1(C(N(CCN(C(c2[nH]cc(C)c2)=O)C)C)=O)CCC(C(C)(C)C)CC1 N1(C(c2cn(C3COCC3F)nn2)=O)CC(O)(C2(CNC(C3CCO3)=O)CC2)C1 Cc1nc(C(=O)NC2(C(=O)N(CCCO)C(C)C)CCCC2)cn1C c1(CC)oncc1C(=O)NC(C)(C(=O)N(C(C)CCSC)C)C1CCC1 CC(C(=O)NC1CCC1NC(=O)C=Cc1ccc(C2OCCO2)o1)C(F)F C(=O)(C(C)CCCC(C)=O)NC(C(=O)N1CCC(OCC#C)C1)CCC c1(C(=O)Nc2cccc(-c3ccoc3)c2)c(C)o[nH]c1=NC(=O)OCC c1(OC)ccccc1C(=O)NC(C)C=CC(=O)NCc1ncccc1C C1(NC(c2c(C)oc(Cl)n2)=O)CCN(C(c2ccc(OCCF)cc2)=O)CC1C c1(NC(C2CCN(CCOCCCCC)CC2)=O)ccnc2ncnn12 Cc1ccc(Cn2cc(C3COCCN3)nn2)c(O)n1 c1(C(=O)NCCC(CC)(C)NC(c2ccsc2C)=O)ccc2c(c1)CC2 C1(c2ccccc2)(CNC(=O)COC(C(C)SC)=O)CCCO1 C12(C(N3CCCN(C(c4n(C)ccc4)=O)CC3)=O)CCCN(C1)S(=O)(=O)C2 C(C)(CNC(=O)CSc1ccccn1)(C(C)C)NC(C(C=CCCC)O)=O CCCC(CCC)=CC(N1CCC(CNC(C2CCCN(CC)C2)=O)C1)=O C(C)(CO)(C(=O)N1CCC(CO)(CNC(=O)COC(C)(C)C)C1)OC Cc1ccc(C(F)CNC(=O)NCC2(C)CC2)cc1F c1(CC(=O)NC2C(C(=O)Nc3cccc(S(C)=O)c3)C2)cc([N+](=O)[O-])ccc1F C(=O)(C1OCCc2c(C)cccc21)NC1CCC(NC(C2(CC)CC2)=O)CC1 c1(C(C)=O)cc(NC2CC(C(F)C(=O)O)C2)ccc1N1CCOCC1 c1(OC)ccc(C=CC(=O)NC2CCN(C(c3ccnn3C)=O)C2)cc1 CC1(C)CC(NC(C2CC(NC(c3cncc(CO)c3)=O)CCO2)=O)CO1 c1(-c2cn(CC(C)NC(C3OCCC3C)=O)nn2)ccc(C(F)F)cc1 Cc1cc(N2CCCNC(=O)C2)nc(NCC2CCOC2C)n1 C1(S(N)(=O)=O)(C(=O)NC2C(CNC(c3n(COC)ncc3)=O)COC2)CC1 CCCCCCC(C)C(=O)NC(C)C(CO)NC(c1cccc(C(F)F)c1)=O C(=O)(C(CC1CCCC1)NC(=O)CC1(C)CC1(F)F)NC(c1nccs1)CC n1(CC(=O)NCC2(CNC(C(CCCC)C)=O)CC2)nnc2c1CCCC2 c1(OC)ccc2c(c1)CC(C)CC2NC(=O)Nc1cccc(CN(C)C)n1 C1(C(=O)NC(C(N2C(C(=O)NC)C=CC2)=O)CO)CN2CCN1CC2 c1(CNC2CC(C(=O)N=c3cc[nH]cc3Cl)(C)C2)ccc(O)c2ccccc12 C1(C(=O)NC23CC(NC(CCC)=O)(C2)C3)CCN(S(=O)(=O)C(F)F)CC1 n1(CC(=O)NC(CNC(c2ccc(C#C)o2)=O)C)nc(C(F)(F)F)c2c1CCC2 C(=O)(C(C(C)NC(c1cncc(C)c1)=O)C(C)C)NCC(=C)Br c1(N2CCCC(NC(C(CC(=C)C)NC(C)=O)=O)C2)ccnc2nc(C)nn12 C1(NC(C=C2CCC(C)CC2)=O)C2CC1N(C(c1cn(CCF)nn1)=O)C2C C1(C(=O)NC2N(C(=O)NCc3cccc(C)c3)CCC2)CN(C)C(=O)CCO1 C(=O)(C(F)(F)CC(=O)N1CCC2(CC2NC(=O)CC(C)O)C1)OC C1(c2nnnn2CCCNCc2c(C)coc2C)(OCC)CC(C)CC(C)(C)C1 C1(CNC(NCC(C=C)(C)C)=NCCC)CCc2nnnn2CC1 C1(C(N2C(CO)CC(NC(C=CC=CC)=O)C2)=O)CC(=O)CC12CCC2 C1(CNC(c2cnn3cccnc23)=O)CC2(CCC2)CN1C(C1CCC=CO1)=O N1(C(CNS(CC)(=O)=O)=O)CCC(O)(CCNC(C2C=CCC2)=O)CC1 c1(CC)cccc(F)c1NC(=O)C(C1CCOC1)NC(c1nsnc1O)=O c1(C(C)C)cc(C(=O)NCC(C)N(C)C(C2CC(OC(C)(C)C)C2)=O)ccc1F C12(CNC(C(C)OCCC=C)=O)CCC1CN(C(=O)CCc1ccncn1)C2 CC1CC(C)N(C(c2cnc3sccn23)=O)CCN1C(=O)C=Cc1ccccc1 CC(CCCCNC(=O)CCC1CCCN1C)NC(C1CC1(F)F)=O C(C(C)C(=O)NCC#CC(=O)NCC(C)N(C)C)OC(C)=O c1(CC(N)C(=O)NC2CC(C(F)CO)C2)ccc(Br)cc1F N1(C(=O)N(CCCO)Cc2ncc[nH]2)CC2CCC(O)CC2C1 c1(CNCC(N2C(C(CCCOC)=O)CCC2C)=O)ccc(C(=O)OC)cc1 C(CCCCC(=O)N1CC(C(F)F)C1)N(C(=O)CC1(O)CCC1)CCO c1(O)cccc(CNCC2N(CC(C)Cl)CC2)c1.c1(CN)cnc(Br)s1 c1(C(=O)NCCN(C(CCOCC)=O)C2CCCC2)cc(Br)sn1 c1(C(=O)OC)c2c(nn1C(C)C)CCC2.c1(OC(F)F)ccc2cc1OCC2=O c1(C(=O)NC(CCNC(CCCCC(=O)NC)=O)C)oc2ccc(Cl)cc2c1C C1(NC(=O)Cc2cc[nH]n2)CN(C(=O)CCCC2CCCC2)CC1CO c1(CC(=O)NCC(C)N(C)C(C2CC=CC2)=O)cocn1 CC(C)CC(C(=O)N1CC(C)CCC1CO)NC(=O)C=CC(=O)OC(C)(C)C C1(C2CCN(C(c3cc(C)c(C)o3)=O)C2)(NC(C(C(CC)C)O)=O)CC1 c1(C(=O)NCCCN(C(C(C=CCCC)O)=O)C(C)C)cccc(F)c1 C1(CNC(c2ncc(N(C)C)nc2)=O)CC2CCC1N(C(c1ccc(F)o1)=O)C2 N1(C(c2c(C)cco2)=O)C2CCC(C2)C1C(=O)NCCC1CCOCC1 c1(CC(C2CCN(CN3CCCC3=O)CC2)C)cnc2c(c1)c(C(C)C)nn2C N1(C(CCS(N)(=O)=O)=O)CCC(C2CC(NC(C3(n4cncn4)CC3)=O)C2)C1 c1(C(C(=O)NCCOC)NC(COCCC)=O)cn(C)nn1 C12(CNC(COCCC)=O)CC(CC)(CN1C(c1cnsn1)=O)C2 C1(NC(C(C)NC(N)=O)=O)(CO)CCN(C(=O)CCC2CC(C)(C)CO2)CC1 C=CCCC(N)C(=O)NC(c1ccccc1O)C c1(OCC)ccc(C(=O)NCC(C)(C)CNC(=O)CCCC(F)F)c(F)c1F Cc1cc(=O)oc(C)c1C(=O)N(C)CCc1cn(-c2ccc3snnc3c2)nn1 C1(CCC(=O)O)(NC(=O)NCC2C(c3onc(C)n3)C2)CC12CCC2 C1(CC=C)(NC(C2CCC(=C)CC2)=O)CCN(C(=O)C=C(Cl)Cl)C1 c1(C(=O)NC(C)CCNC(C2(C(C)(F)F)CCOCC2)=O)occ2c1CCOC2 S(=O)(=O)(c1cnc(NC2CCCn3nccc32)c(Cl)c1)N1C(C)C(CO)CCC1 C1(NC(C(CSC)(C)C)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)c(F)c1)C C(=O)(C(F)(CNC(C12C(=O)C3CC1C2C3)=O)C(C)C)N1CC(OC)C1 N1(C(C(=O)NC2CC(C(=O)OC(C)(C)C)C2)=O)CCCCC1c1ccc(CN)o1 C1(NC(COCC=C)=O)CC(OC)CN(C(=O)C(COC)OCC=C)C1 C1(N2CCOCC2)(CNC(=O)NC(CN(C)C)C2CCC2)CCCC1 C1(CC=C)(NC(C2CC=CCO2)=O)CCCN(C(c2n[nH]cc2Cl)=O)C1 C1(NC(CSC)=O)(CNC(c2cccc(C)c2F)=O)CC2CCC1C2 CC(C)(C)CCCCC(=O)N1CC2C=CC1C(C(N1CC(c3ccon3)C1)=O)C2 C12(C(C)C)CC(C1)COC2=O.C12CC1NC(=O)C(=O)N2.C(=O)OC.C1CC1.O(C)C N1(C(c2nc(OC)c(C)s2)=O)CCCC(C2(NC(=O)C(C)N(C)C)CC2)C1 c1(SCC(=O)NCCNC(C23CCCC2(CO)C3)=O)cccc2cccc(Cl)c12 CN1CC(C)(C)CC1C(=O)NCCC1(NC(=O)C2=COCCC2)CCC1 C#CCCCCCC(=O)NC1CCC(N(C(=O)COCc2nc(CC)no2)C)C1 Cc1ccc(C(=O)NCC2CC2NC(=O)C(F)(F)C2CC2)cn1 c1(C(=O)OC)coc(C=CC(=O)NCC(C2CCCCO2)N(C)C)c1 C(=O)(C(C(C)C)n1cc(Br)cn1)N(CCNC(CSC)=O)C1CC1 N(C1CCc2ccc(F)cc21)CC(C)CO.CO C1(C(=O)NC(C(C)C)C(=O)OC(C)(C)C)CC12CCCCC2.C1(C)C(=O)N1 N1(C(C2(OC(C(=O)NC)OCC)CC2(C)C)=O)CCOC(CCO)C1 c1(C(=O)NC)cccc(C(N2CC(C(C)NC(=O)C(=Cc3cn[nH]c3)C)C2)=O)c1 c1(C(C(=O)NCCCSC)(C)N(CCOCCO)C(C)C)ccc(Cl)cc1F c1(NC(C2CC2C2CC2c2ccccc2)=O)cc(F)ccc1Cl C1(CC=C)(C(=O)NC(CO)C(C)C)CCCN1C(=O)CCCOC C1(OCCNC(CN(C)C)=O)CC2C(C1)C2(C)C c1(CC)cn(C)nc1C(=O)Nc1cccc(NC(=O)CCC2CCCCC2)c1 C1(CC)CN(C(c2cc(C3CC3)cc(F)c2)=O)CCN1C(=O)C(C)OCOC c1(C(CNC(c2c(C)scn2)=O)NC(C2CCOC2)=O)ccccc1Br c1(N(C(COCC)C(=O)NC(c2nc(C3CC3)cs2)C)C)cccc(F)c1Cl C1(C(=O)NC2(CN(C(=O)C=Cc3cccc(CO)c3)C)CC2)COCCC1(F)F Cc1nc(SCC(=O)NCC(CO)NC(=O)CCc2ccnn2C)n[nH]1 Cc1nccnc1C(N1CC2C(CNC(C3C=CCC3)=O)C2C1)=O c1(NCC2C3CN(C(C4C(C)CC5CC5C4)=O)CC32)ncccc1[N+](=O)[O-] C12(NC(CCc3c(C)ncs3)=O)CCC(C1)N(C(=O)CC1(C)CCCO1)C2 c1(NCSC(F)(F)F)cc(Cl)nn2cnnc12 CC1CN(C(=O)C2=NOC(C)(C)C2)CC(C)N1C(c1ccc(F)cn1)=O c1(CCC(N2CC3C(N(C(C(C)SC)=O)C)C3C2)=O)ccc(Cl)c(Cl)c1 N1(C(c2c(CC)scc2)=O)CCC=C(C(=O)N(CC(F)F)C)C1 C1(C(=O)NCCOCCN(C)C(c2ccncc2)=O)CCOC1C(F)(F)F Cc1nn(C)c(C)c1CN1CC(O)(C(=O)NC2CCC2N2CCCC2)C1 Cc1cc(C(N2CC=CC(NC(=O)C3=CCS(=O)(=O)C3)C2)=O)c2c(C)n[nH]c2n1 c1(N2CCC(CNC(c3cnc(C4CC4)[nH]3)=O)C23CC3)ncnc2c1CCCC2 N1(C(c2nc(N(C3CC3)C)oc2)=O)CCCC(CCC(=O)N(CC(C)C)CCC#N)C1 C1(COC)(OC)CCCN(Cc2nnc(C3CCOCC3)n2CC2C(C)C2(F)F)C1 c1(OC)cc(OC)cc(C(=O)NCCOCCNC(=O)C2=CCCSC2)c1 N1(C(=O)CCC2CCCCC2)CCCC(C2CCCN(CCC3CCOC3)C2)C1 Cc1cnnc(O)c1C(=O)NC1CCN(C(=O)C(O)CC(C)C)C1 N1(C(c2sc3c(c2)CC(C)CC3)=O)CCC(C2CCCN(C(C3CCCO3)=O)C2)C1 N1(C(CNC(N)=O)=O)CCC2(CNC(=O)CCCCC(F)(F)F)CCCCC12 C1(CC(C)C)(C(=O)NCC2CC2CNC(c2ccc(CO)nc2)=O)CCNC1=O c1(N2CCC(CCNC(=O)CNC(C3CCOC3)=O)CC2)ccc([N+](=O)[O-])cc1 C1(NC(C(CC=C)(F)F)=O)CN(C(c2cc(Cl)c(N)cc2)=O)C2CCCCC12 C=CCC(CC(F)F)C(=O)N1CCC2C(CCN2C(C2CC(SC)C2)=O)C1 c1(NC(C2CCC(NC(CCCOCC=C)=O)C2)=O)cc(CC)cc(C)c1 c1(-c2ccc(CN(C3CN(C(=O)NC(CC)(C)C)C3)C)o2)cccc(Br)c1 N1(C(c2cc(OC)cc(C)c2)=O)CCCC2(CCC2NC(=O)CCOC(C)=O)C1 N1(C(c2ncn(CC)n2)=O)CCSCC1C(=O)NCCc1cccc(F)c1 N1(C(CC2ON=C(CC)C2)=O)C2CCC(C2)C1C(=O)N(CC(C)(C)C(F)(F)F)CC c1(C(=O)NCC2(F)CC(CNC(COCCC)=O)C2)ccc2ccn(C)c2c1 C1(C(=O)NCC2(CNC(c3cc(C(F)F)ccn3)=O)CCC2)COCCC1(F)F c1(C(=O)NC(CCNC(CC(C(=C)C)O)=O)C)c(C)nn2cc[nH]c(=O)c12 c1(C(=O)OC)cccc(CN2CCSCC2C(=O)NCCCCSC)c1 c1(COC)noc(C(N2CC(CNC(c3cnc(C)[nH]3)=O)C2)C)n1 C1(C)(NCCNC(NCC2(OCC)CCCSC2)=NC)CCOC2(CCC2)C1 C1(O)CC2CC(C(=O)NCCc3ccc(C4CC4)cc3)CC12.C1(=O)CN1.CCNCC N1(C(CCOc2cccc(C)c2)=O)CC2CC1CCN2C(C1CCCSC1)=O N1(C(CC2C(C)(C)C2)=O)CCCCC(NC(C2C=CCS2)=O)C1 C1(NC(=O)C(c2ccc(Cl)cc2)O)CC2(C1)CN(Cc1cccc(Br)c1F)C2 c1(N(C)CC2CCCO2)nc(N2CCN3CCCC3C2)c2c(n1)CCS2 O=C1CCC(C(=O)N2CC(NC(=O)Cc3nc[nH]n3)C(O)C2)c2ccccc21 c1(C(=O)NCC2CN(C(C(C)C3CC3)=O)C(C)C2)ccc(C(C)(F)F)nc1O C(=O)(CCCCC(=O)NCC1CC1NC(=O)C(F)(F)c1cnccn1)OC C(=O)(N1OC2C=CC1CC2)C1C(CNC(=O)CCc2cncs2)C1 C12(NC(c3c(C)ccc(C)n3)=O)CCCC1N(C(=O)CSCC(N)=O)CCC2 C#Cc1ccccc1CC(N1CCCC1C(=O)NCC=CBr)=O c1(CC(=O)NC(C2CCN(C(c3ccc(Cl)nc3Cl)=O)C2)C)cccc(N)c1N C1(C(=O)NC(C2CN(C(C(C(C)C)N(C)C)=O)C2)C)CC12CCCCC2 Cc1cc(F)c(CC(N2CC(F)CC2CNC(=O)C(C)C(F)F)=O)cc1F N1(C(=O)Cn2cccc2)CCOCC1CCNC(C1(n2cccn2)CCC1)=O CCC(C)(COC)CNC(=O)CC1(CNC(C2(C)CCCC2O)=O)CC1 N1(C(C2(N=[N+]=[N-])CC2)=O)CCN(C(c2sccc2Cl)=O)C2CC12 C1(NC(CNC(C)=O)=O)C2COCC1CC(NC(c1c(C)ncnc1O)=O)C2 c1(C(N(CCC(N2CCC(CC)C2)=O)CC=C)=O)cncc(OCC)n1 c1(C(=O)NC(C)C(C)NC(c2coc(CO)c2)=O)cc(S(N)(=O)=O)c[nH]1 c1(CC)cc(CN2CC(C(N3CCOC4CC34)=O)C2)ccc1C N1(C(CNS(NC)(=O)=O)=O)CCC2OCCN(C(=O)CC3(OC)CCC3)C2C1 C(=O)(C(F)C(C)CNC(C1CCC1OCC)=O)NCC1CCC(=C)CC1 Cc1cc2c(C(=O)N(CCC(C)NC(=O)C(C)CC3CC3)C)nccn2n1 N1(C(c2cc(C(C)C)nn2C)=O)CC(C)(C)OCC1CNC(c1ccc(Cl)o1)=O c1(C(=O)NCCN(C(C2(S(C)(=O)=O)CC2)=O)CC)ccc(Cl)c(OC)c1 C1(C#N)(CC)CCN(C(C2(CC)CCN(C(=O)C(C)OCC(C)C)C2)=O)CC1 C(=O)(CCCCCCC)N1C23CC1(C2)C3.C=CC(CC(=O)OC)OC CC1CC(NC(=O)C(F)(F)F)CN(Cc2ccccc2CCC(=O)O)C1 c1(C(=O)NC2CN(C(c3c(CC#N)cccc3)=O)C2)cc2ccncc2c(O)n1 C1(N(C(C2(C(F)F)CC(=C)C2)=O)C2CC2)CCCN(C(=O)C=Cc2ncc[nH]2)C1 c1(COCC(=O)N(CC(CC)NC(=O)CC2(C)CCCO2)CC)ccncc1 N1(C(=O)Cn2cccc2)CCOCC1c1cn(CCF)nn1 C1(C(=O)NC2(CNC(c3noc(CC)c3C)=O)CCC2)CCc2n[nH]c(C)c2C1 N1(C(CC=CC)=O)CCn2ncc(S(C)(=O)=NC(=O)C3(CC)COC3)c2C1 Cc1cc(=NC2CCN(C(=O)C3CC3)C2)[nH]c(N(C)Cc2cncs2)n1 c1(NC(C)=O)cc(C(=O)N(C2CN(C(C3CC3(F)F)=O)CC2(C)C)C)ccc1F C1(NC(Cc2c(C)ncs2)=O)CCN(C(C2CN(S(N)(=O)=O)C2)=O)CC1C N1(C(C2CCN(CC)C2)=O)CCC2C(NC(c3cnc(C)s3)=O)C12 c1(C(N2C(C)(CC(=O)NCc3c(C)c[nH]n3)CC2)=O)cccn(C)c1=O C1(C)(CNC(c2c(C(=O)OC)c[nH]c2)=O)CCN(C(c2ccc(Cl)s2)=O)C1 CC1C(O)CCCN1C(C12C(NC(c3cnn(C)c(=O)c3)=O)C3CC1C2C3)=O c1(C(N2CC(O)(CCNC(=O)CC34CCCC3C4)C2)=O)ccc([N+](=O)[O-])cc1 CCCCCC(O)C(=O)NC(CNC(=O)CCNC(=O)C=CCl)CO C1(C(N2CCCC(CNC(C3C(C)(C)C3)=O)CC2)=O)CCCC2CCCN12 n1(CC(=O)NCC(C)NC(C2(O)CCC(C)(C)CC2)=O)nc2ccccn2c1=O c1(C(=O)NC2CC(CNC(c3[nH]n(C)c(=O)n3)=O)C2)cc(F)ccc1C(F)F c1(NC(C2CCC(CCCC)CC2)=O)ccc2c(c1)CC(C)(C)O2 c1(CN2C(C(=O)NC(CC)C(F)(F)F)CC3CC32)cccc(Cl)c1F N1(C(COCC)=O)CCCC(C2CCCN2C(=O)CCOC)C1 c1(C(N(CC(C)N(C(CCOC(C)C)=O)C)C)=O)cnoc1C1CC1 c1(SC)ccccc1C(=O)NC(C)C(C(C)C)NC(c1sc(=N)[nH]c1C)=O C(=O)(CC1=CCCC1)N(C1CN(C(=O)CCCSCc2cccs2)CC1F)C Nc1cc(F)cnc1C(=O)NCC1(O)CN(C(c2[nH]nnc2C2CC2)=O)C1 N1(C(C(C=C)OC)=O)CCCN(CCNC(=O)C(C)OC)CC1 C1(F)(C(=O)NCC2N(C(c3cc(C(N)=O)on3)=O)CC2)CCOCC1 C1(NC(CN(CCC#C)C)=O)CCCCN(C(c2cccc(C(C)C)n2)=O)CC1 N1(C(C(C)OC)=O)CC2COCCC2(NC(c2cc(Br)ccc2C)=O)C1 N1(C(c2cnc(O)cc2O)=O)CCC2C1CCCN2C(c1ccc(Cl)cc1Br)=O N1(C(=O)C(F)=CC2CC2)CCN(CCNC(=O)C(F)(F)c2nccs2)CC1 CCC(O)CC(=O)N1CC(CC(C)NC(C2(O)CCOCC2)=O)C1 N1(C(c2cc(COC)sc2)=O)CCN(CCNC(=O)CC2CCC(=O)NC2)CC1 N1(C(=O)C2=C(Cl)CCCC2)CC(NC(=O)C=CC2CCC2)CC12CCCCCC2 C(=O)(CCCCCN=[N+]=[N-])N(CCC(=O)NCC12COCCN1C(=O)COC2)C C1(C(=O)NCC2(NC(c3[nH]c(=NCC)sc3)=O)CCCC2)CC12CCCCCC2 C#CC1(CNC(=O)C(O)CNC(=O)C(C)(O)CCN(C)C)CCOCC1 c1(C(N(CC(C)NC(=O)CC2CCC(F)(F)CO2)C)=O)nccc2ncncc12 CC1=C(C(=O)NCC2C(CNC(c3csnc3C)=O)C2(F)F)CCCC1 N1(C(=O)CC2C=CCC2)CCC2(CCN(Cc3ccc4c(c3)COCC4)C2)C1 CC1C(NC(=O)COCc2ccccc2)CCN1C(c1cc(C2CC2)on1)=O C1(C(=O)NC(C)CNC(c2cn(Cc3cccs3)nn2)=O)CCCS1(=O)=O c1(C(=O)NC2CN(C(C(CCC)CCC)=O)C2)cncc2c(OC)cccc12 C1(C(=O)NC2(C)CN(C(C3C(C4C(C)C4)C3)=O)C2)COc2ccccc2O1 Cc1ccc(NC(C2C3CN(C(c4ccc(CO)c(Cl)c4)=O)CC23)=O)c(C)c1Br c1(C(=O)OCC)cc(-c2nc(C(C)COC)no2)nc2ccc(C)cc12 C12(C(=O)OC)CCCC1N(C(=O)C(S)C(C)C)CCC2 CN1CCCC(C(=O)NCc2ccc(C(=O)NCC#CCCO)cc2)C1 N1(C(CSCC(C)C)=O)CC2CC(NC(=O)CC(O)C3CCCC3)CC1C2 N1(C(CCOCCC)=O)CCC(C(N2CCC(OC3CCC3)C2)=O)CC1(C)C C(=O)(CC1=CCN(C)CC1)N(C1CCN(C(C(C)NC(c2cccs2)=O)=O)C1)C CN1CCCC1(C)C(=O)NCC1CCCCC1NC(c1cc(Br)cn1C)=O CCCCC(C(=O)NC1(C)CN(C(=O)C=Cc2ccoc2)C1)C(C)C C(CC(O)CNC(c1cn(-c2ccccc2)cn1)=O)NC(c1ccon1)=O CCCCC(CC)CCC(=O)NCC1CN(C(=O)C(F)(F)C(C)O)CCO1 C1(NC(C)=O)CCC(CNC(=O)Cc2ccc(-n3ccnc3)cc2)CC1 C1(C(=O)OC(C)C)CS(=O)(=O)CN1C(c1cc(-c2ccccc2)cs1)=O N1(C(c2c(Cl)ccc3c2OCO3)=O)CCc2cc(F)cc(Cl)c2C1 C(=O)(CCCCC(N)=O)NCCCC(C)NC(C1CCN(S(C)(=O)=O)CC1)=O CCCCCC(O)C(=O)NC(C)CCNC(c1ccc(OCCOC)c(F)c1)=O C1(NC(C(=O)NCC)=O)CCN(C(c2ccc(N(C)C)nc2)=O)CCC1SCC CCCC(C)(CC)C(=O)N1CC(NC(=O)C=Cc2n[nH]c(C)n2)CCC(O)C1 C1(CC(=O)NCc2nocc2C(=O)NCC2(Cl)CC2(F)F)CCCCC1 C1(C(N(CC(C)NC(COCCC=C)=O)C)=O)CN(C)C1 c1(OC)ccc(NC(=O)C(C)N(C(=O)CC2CC=CCC2)C)c(C)c1 C1(C(N(C)Cc2cn(C)nn2)=O)CCN(C(=O)C2=COCC2)C1(C)C C1(C(=O)NC2CC(C)(NC(c3cnc(C(C)C)n3C)=O)C2)C2CS(=O)(=O)CC12 c1(C(N(CCCCCNC(C2CC(C#N)C2)=O)C(C)C)=O)cc(Cl)c(Br)[nH]1 c1(-n2c(CC34CCCC3C4)nc(CCCO)n2)ccc2ccccc2c1 N1(C(c2c(C(C)C)n[nH]c2)=O)CCCC(C(C)(O)CNC(c2occc2Cl)=O)C1 CC1CN(C(=O)CCCC2CCCC2)CC(C)C1NC(c1ccnc(F)c1Cl)=O N1(C(C2C(C)(C)OC(=O)N2)=O)C2CC=C(C(=O)NCCCN3CC=CC3)C1CC2 C(=O)(C(O)C(C)(C)C)N1C(CN(C)C(c2nscc2N)=O)CCC1 CCC(C(=O)NC1CC12CC(C)(NC(=O)OC(C)(C)C)C2)C(C)C CCC(C)(C)CC(=O)NCC1(F)CCC(NC(=O)C(O)Cc2cnc[nH]2)CC1 C=CC1(CC(=O)NCC2(C)CCN(C)C2)CN(C(c2sc(F)cc2C)=O)C1 C1(C(=O)NCC2(C(F)F)CCN(C(C(CC)SC)=O)C2)CC2C(C1)C2(C)C c1(NC(C(N2C(CCNC(c3cc(Cl)c[nH]3)=O)CCC2)=O)=O)ccc(Cl)c(F)c1 C#Cc1cc(NC(=O)C#CCNC(=O)C2=C(Cl)CCOC2)cc(F)c1 c1(C(=O)NC(C)CNC(c2ccc(F)cc2F)=O)ccn2c1CCCC2 CCC(CC)C(F)C(=O)N1CCCC1C(C)(C)C(=O)NCc1cc(OC)ns1 C1(CCNC(C(C)(C)CO)=O)CN(C(C2Cc3ccccc3S2)=O)CCS1(=O)=O c1(OC(C(=O)NCCNC2CCSCC2)F)ccc(Cl)c(F)c1 C1(C(=O)NC(C2CCCCC2)CC)CCCCN1C(=O)Cc1ccc(C)o1 Cc1cnc(NC(=O)Nc2cc(-c3cccnc3)nn2C)c(Br)c1 C(C)(CN=c1[nH]ccn2c(C(C)(C)C)nnc12)NC(=O)NCc1cccc(C)c1 C1(c2nnnn2C2CCC2)(NCc2ccc(OC)c(F)c2)CC(C)NC(C)C1 c1(C(=O)NCC(C(=O)OC(C)C)F)c(Cl)ccc2cccnc12 c1(C(=O)NC2CN(C(c3cnn(CC)n3)=O)C(C)CC2)cc(O)c(F)cc1N C#Cc1ccc(C(=O)NC2CN(C(c3cc(C)cc(Cl)c3)=O)CC2C)cc1C C1(NC(c2c(COC)noc2)=O)CN(C(c2cccc(F)c2)=O)CC1S(C)(=O)=O N1(C(C=NOC)=O)CCC(c2ccccc2)(NC(C2CC2COC)=O)CC1 C1(CC=C)(NC(c2oc(CC)nc2C)=O)CCN(C(=O)COCC)C1 c1(OC)cc(NC(C2CC23CN(Cc2cc[nH]n2)C3)=O)c(F)cn1 N1(C(C(C)(C)S(C)(=O)=O)=O)CCC2(CCC2)C(CNC(=O)C2=CCCOC2)C1 Cc1cc(CNC(C2(CCNC(C3(F)CC=CC3)=O)CC2)=O)ccc1F C1(F)(CNC(c2ccc(C(F)(F)F)[nH]2)=O)CCN(C(c2cccs2)=O)C1 N1(C(CCCNC(N)=O)=O)CCC(NC(=O)CC2CCC=CCC2)C(CO)C1 c1(C(=O)NC(C(=O)NCC2(C(C)(C)OC)CC2)CC(C)C)cc2ncccc2[nH]1 c1(C(N2C3CN(C(C4(F)C(C)(C)C4(C)C)=O)C(C3)C2)=O)ccc(O)cc1[N+](=O)[O-] c1(CNC(=O)NCc2cc(C3(CO)CC3)[nH]n2)ccc(C2CC2C)o1 C=CCC(C(=O)N1CCCN(C(c2[nH]cc(COC)c2C)=O)C(C)C1)C(C)C N1(C(C2N(c3nc(C)c(Br)cn3)CC(O)C2)=O)CCCC(C)(O)CC1 C1(NC(C(C)(C)c2cccnc2)=O)CCC(Nc2ncc(F)cn2)CC1 CC1CN(C(=O)CC2CC3(CCO2)CC3)CCN(C(C2CCCC2F)=O)C1 C=C=CCCC(=O)N(CCCNC(=O)C(n1ccc(Br)n1)C)C Cn1c(C(=O)NC2CC(O)(CNC(C3CSCCS3)=O)C2)cc2ccccc12 CC1(CC(=O)NCCCCO)CCN(C(=O)C2=CCSC2)CC1 N1(C(=O)Cn2ncnn2)CC2(CCN(Cc3ccc(Br)cn3)C2)C1 C12(CC)COC(C(N3CCCC(NC(=O)C(C4CCCCC4)O)C3)=O)(C1)C2 C1(CC=C)(C(=O)N(CC(C)COC)C(C)C)CN(C(=O)CCc2cc(C)[nH]n2)C1 N1(C(C2(C)N(C(C3C(C(C)=O)COC3)=O)CCC2)=O)CC(C)OCC1C N1(C(C2CCC(=O)NC2)=O)CCCC(O)(CNC(C2(O)COC2)=O)C1 c1(COC)ccc(Cl)cc1Cl.N12CC=CC1C(C)(C)CNC(=O)NC1C(C1)C2=O c1(C(N2CCC(C)(CNC(C3(O)COC3)=O)C2)=O)cc2ccc(Cl)cc2[nH]1 C1(CC(=O)N(CCCNC(=O)C=CC2CCCO2)C)CC2(CCOCC2)CO1 C#Cc1ccccc1CC(=O)N(C1CCCCN(C(=O)C(C2CC2)OCC)C1)C c1(C(=O)OCC2(CC=C)CCOCC2)ncnc2c1CCCC2 C1(C(N2C3(CNC(=O)Cc4csc(C5CC5)n4)CC(C2)C3)=O)Cc2cscc2C1 C1(C(=O)NC(C(=O)NC(C2CCOC2)C#C)Cc2cn[nH]c2)CCC(C)(C)CC1 c1(C(=O)NC(CCCNC(COCCOCC)=O)C)ccc(C2CC2)cc1Cl n1(CC(=O)NCC2C(C(=O)OC)C2)ncc(=O)c2ccccc12 C1(CNC(c2c(C)ncn2C)=O)CCC12CCN(C(C1CC(C)(C)O1)=O)CC2 CC1CCC(C)N1CC(=O)NCC1CC(NC(=O)C(C)OCC2CCCO2)C1 C12(C(N(CC)Cc3cnn(C)c3)=O)CC(CO)(CN1C(c1nccn1CC)=O)C2 C(CC1=CCN(C(c2[nH]nc3ncccc23)=O)CC1)NC(C1CC12CC2)=O c1(OC)ccc(OC)c(CC(=O)NC2CN(C(c3ccn(CC(F)F)n3)=O)C2)c1 c1(-c2c(C)ccs2)ccc(C(=O)NC2(CO)CCC2)c(C)n1 C1(C(ONC(=O)Nc2cccc(C#N)c2)C)CCCN1NC(=O)C1CCOC1C=C c1(OCC)ccc(Cl)nc1C(N1CCN(CC(C)NC(C2CCC2C)=O)CC1)=O C1(C(C)CNC(C2CCOCC2)=O)CCN(C(=O)C(C)(C)C2CCOCC2)CC1 Cc1ccc(C)c(CN(C2CN(C(=O)C(C)n3ccnc3)C2)C)c1 C1(C)(CNC(c2scc(CCCOC)n2)Cc2nnnn2C(C)C)CCCOC1 c1(C(N(C(CNC(C(C)OCCOC)=O)C2CC2)C)=O)c(OC)cccc1OC Cc1cc(N)cc(C(N2CCN(C(c3cccs3)=O)CC(CO)C2)=O)c1F C1(C(=O)NC(CC#C)CO)COCCN1C(C1CS(=O)(=O)C1)=O N1(C(C2(CNC(=O)C3CC3)CC2)=O)CCC(C)(C)C(NC(c2ccc(Cl)s2)=O)C1 C1(C(N(C)C)=O)C2CC2CN1C(=O)CN(C)C(c1cncn1C)=O C(=O)(CN=C(NCc1cc(Br)cs1)NC(c1ccc(Cl)cc1)C)NCC N1(C(c2cnc(C(C)=O)s2)=O)CCC(NC(c2cn3cccnc3n2)=O)C(C)(C)C1 C1(CNC(C23OCC(COC)(C2)C3)=O)COCCN(C(C2CCCC2)=O)C1 c1(C(=O)NC23C(CN(C(C(CC(C)C)N(C)C)=O)C2)C3)cc2c(s1)CCOC2 c1(C(N2CCN(C(=O)C3=CCSC3)CC2c2ncc[nH]2)=O)ccc2nc[nH]c2n1 c1(C(=O)NC2(C(NOCCC(=C)C)=O)CC(O)C2)cc(O)nc(C)n1 C1(C(=O)NCCCn2ccnn2)(CNC(C2C(CCC)C2)=O)CC(C)(C)C1 c1(C(N2CCC(C)C2C(=O)NC2CC(O)C(O)C2)=O)ncc2ccccn12 C1(NC(=O)COC(F)F)CCCCC1NC(C1(n2cnnn2)CCCCC1)=O c1(CC)ccc(C)c(NC(=O)NCc2ccc(Br)nc2)c1 N1(C(C)C)CC(C(=O)NC2(CO)CCCN(C(C3(C4CC4)CC3)=O)C2)CCC1=O C(CC(CC)C(=O)N1CCC(N(C)C(c2ccc(=N)[nH]n2)=O)C1)=CC N1(C(C(CCC)CC)=O)CCC(CCNC(=O)C(C)(C)COC)C(F)(F)CC1 c1(OCC(N2CCC(CNC(CC=C)=O)C(C)(C)C2)=O)ccc(S(N)(=O)=O)cc1 N1(C(CCC2N(C(c3cc(SC)oc3)=O)CCC2)=O)CC2(CSC2)C1 C(=O)(CCCC(=O)NC1(CF)CCN(C(=O)CCCOC)C1)N(CCC)C(C)C Cc1nnnn1CC(N1CCCC1CC(=O)NC(c1ccncn1)C)=O n1(CC)nc(C(=O)NCC2CCN(C(=O)C(C3CC3)SC)C2)c(C)n1 C(=O)(C(CN=[N+]=[N-])NC(=O)CN=[N+]=[N-])NCC(c1nncn1C)C N1(C(C2CC(OC)OC2OCC)C(=O)NC(CC)C)CCC2(CCCCO2)C1 C1(C(=O)NC(CNC(CC2C(C)(C)CCCC2)=O)CO)CC2(C1)CC1(CC1)C2 N1(C(c2cc(C)n(C(F)F)n2)=O)CC2CN(C(c3cscc3C(F)F)=O)CCC12 C1(O)(CCNC(C2CCC2(F)F)=O)CCN(C(c2ccncc2O)=O)CC1 c1(C(C(=O)NC(C)CN(C)C(C2CCN2S(C)(=O)=O)=O)(F)F)ccc(Cl)cc1 c1(N2CC(C)(CC)OCC2)nc(N2CCC(OC(C)C)C2)c2c(n1)CCCCC2 C(=O)(C(C)NC(=O)CC1(NC(C2CC2(C)C)=O)CCC1)NC(CC)C C1(NC(Cc2cc(C)ns2)=O)CN(C(C2CNC(=O)N2)=O)C2(CCCCC2)C1 C(=O)(C1CCCc2cncn21)NCCCC(C)NC(c1nn(C(F)F)cc1Cl)=O c1(C(N(CC(CC)O)CC)=O)ccnc(CNC(=O)CC(CC)OC)c1 N1(C(C(C=C)O)=O)CC2(C1)C(NC(c1ccn(CC)c(=O)c1)=O)CCS2(=O)=O C(=O)(C(C)C(C)NC(C)=O)NCC(COC)(F)F N1(C(C=C(C)C(F)F)=O)CCC(O)(CNC(C2COCCN2CC(F)F)=O)CC1 CC1C(CC(=O)NCC(C2CC2)NC(=O)C=CCN(CC(F)(F)F)C)C1(F)F Cc1cnc(C(N2CCCC(CC(=O)NC(c3ccc(O)nc3)C)C2)=O)cc1C C1(NC(C(CC#C)NC(=O)C(O)CN(C)C)=O)CN(C)CC1(C)C N1(CCC)CCCCC1C(=O)N(C1CCCC1)CCNC(C12CCC(C1)C2)=O N1(C(C(=O)NC(C)C)=O)CC2(CCC2NC(=O)C(C)CN(C)C)C1 c1(N(C)C)ncc(C(=O)NC2(CNC(=O)C=Cc3cnc[nH]3)CCC2)s1 CC1CC(C)CN(C(=O)CN2CCCC(CCNC(C3(CN)CC3)=O)CC2)C1 N1(C(C2(CC=C)CC2)=O)CCCC(N=C2N=C(C)Nn3cccc3N2)(CO)C1 c1(N(c2ccncn2)C(=O)NCC(CC(=O)O)C2CCC2)ccc(Br)c(Cl)c1 c1(NCC(CC)C(C)(F)F)[nH]c(=NCC2CCC23CCC3)nc2scnc12 C(=O)(C1CCCc2n[nH]cc21)NCC12CN(C(c3c(CC)c[nH]n3)=O)C(C1)CO2 C1(CNC(C(C(C)C)SCC)=O)CN(C)CCN1C(c1cn(C2CC2)nn1)=O c1(CC(N2CCC(NC(=O)COC(F)(F)F)C(O)C2)=O)c[nH]c2ncccc12 CC1(C)CC(NC(=O)CN=S(C)(C)=O)CN1C(C1CC2(CSC2)C1)=O c1(C(N2CCCC(CN(C(C(C)OCC=C)=O)C)C2)=O)n[nH]c2ccc(Cl)cc12 C1(C(=O)NCC(C)(C)CNC(=O)C(F)F)(OC)CCC(c2ccccc2)CC1 C(=O)(CC(C(F)F)NC(c1nc(Cl)oc1C)=O)NCCN(OC)C c1(CN2CCC(NC(Cc3nc(C)oc3)=O)C2)ccc(Cn2ccnc2)cc1 c1(C(N(C(CNC(c2c(OC)cnc(Br)c2)=O)C)C)=O)cccc2[nH]ncc12 C(CCC(O)C(=O)NCC(C)F)NC(C(C)SCCCC)=O CC(C)CCC(F)C(=O)N1CCCC(CNC(=O)CN(C(=O)C(C)C)C)C1 c1(OC)cc2cc(C(=O)NC(C)C(C)NC(c3n[nH]cc3Cl)=O)[nH]c2cc1OC C12(CC)CC(CNC(=O)Cn3cc(CC(C)O)nn3)(CN1C(c1cocn1)=O)C2 c1(C(N2CCC3CCCCC23)C(=O)NC2(C)CC2)cc(Cl)c(Br)c(Cl)c1 CCC(C(=O)NCCN(C)C(C1(C(=O)N(C)C(C)C)CC1)=O)C(F)(F)F C(c1cn(C)c2ccccc12)=C1CCN(C(C(=O)C(CSC)=O)C(C)C2CC2)CC1 Cn1nc(C(=O)NC2CC3CN(C(c4ccc([N+](=O)[O-])s4)=O)CC23)c(Cl)c1Cl C1(C(N(C)CCC2CCCN2C)=O)(CO)CCN(C(=O)C(C)(C)c2ccno2)C1 N1(C(CC(CC)SC)=O)CC(NC(=O)COc2cccc(F)c2)CC1(CC)CC c1(C(=O)NCC(C)(CO)NC(c2cn(C)nc2Br)=O)noc2c1CCCC2 N1(C(C(CCC)O)=O)CCN(C(c2occc2Cl)=O)C(CF)C1 CN1CCCC2CN(C(=O)NCC3CCC3c3cccc(Br)c3)CC12 C(=O)(C1=NOC2(CCC2)C1)N1CCC(F)(CNC(c2c(C)csc2Cl)=O)CC1 Cc1nccc(N(C(C)CNC(C2CC(=O)N(c3cnn(C)c3)C2)=O)C)n1 c1(NC(C(Cn2cccn2)NC(c2c(NC)cnnc2)=O)=O)cc(F)ccc1C [N-]=[N+]=NC1CCC(C(=O)NCC2(NC(=O)Cc3cc[nH]n3)CCCCCC2)CC1 c1(C(=O)NCC2C(C(N(CC(CCC)O)C)=O)CCC2)cnc(O)c(C)c1 N1(C(CC2(OC)CCCC2)=O)CC(C2CN(C(=O)C(C)(O)C3CCOCC3)C2)C1 N1(CC(N2CC(NC(C(C)SCC)=O)C2)=O)C(=O)C(=O)N(C)C1=O N1(C(C(C)(C)CF)=O)CCC2(CC1)CN(C(C1CN3CCCC1C3)=O)C2 C(=O)(C(C)(C)CCNC(=O)CN1CCC(O)CC1)N(C(C(C)SC)C)C c1(SCC(=O)NCC(CC)NC(c2c(C(C)C)cnn2C)=O)ccc(C)c(C)c1 C1(CNC(C2CC3CCC2C3)=O)CC2CCC1N(C(=O)C(F)C1CCOC1)C2 c1(C(N(C2CCN(C(c3nccn3C)=O)C2)C)=O)cc2oc(Br)cc2s1 c1(C(N(C2CC(NC(CCc3ccc(CC)cc3)=O)C2)C)=O)ccnc(F)c1N c1(CC)n[nH]c(CC)c1CC(=O)NC1CN(C(=O)CC2(C)CC2)CC1OC c1(OC)cc(N)c(C(=O)N(C2CN(C(C3CCC3C)=O)C2)C)c(Br)c1 c1(C(C)(C)NC(C2CC(CNC(=O)CCN3CCOC3=O)C2)=O)cncnc1O C12(C(N(CC(C)(CO)CO)C)=O)CC(CO1)N(C(C1CNC(=O)N1)=O)C2 C12(NC(C(C)OCCC(C)C)=O)CC1CN(C(C1(O)CCSCC1)=O)C2 CC1CCC(NC(=O)CCc2cc[nH]n2)CN1C(=O)CCCc1cnn[nH]1 C1(CNC(c2c(C)n(C)nn2)=O)CN(C(=O)Cc2cccc(C(F)F)c2)CC12CC2 C(=O)(C(O)C1=CCCCC1)NCC(C(N1CC(OC)C2(C1)CC2)=O)O CC1CC(c2ccc(C3CN(C(=O)CSc4nncn4C)CC3C)cc2)CCO1 c1(SC(C(=O)NCC(CC=C)NC(c2csnn2)=O)C)ccccc1Cl N1(C(c2c(C(C)=O)cn(C)n2)=O)CC2CCC1C(NC(=O)C(C)C#N)C2 C12(NC(C3CCCC(C(=O)OC)C3)=O)CCCN(C(c3cc(C)sn3)=O)CC1C2 C#CC1(C(=O)NC(c2nncn2C)CO)CN(C(C2CCO2)=O)C1 C12(C(N3CCC(OCC(=O)NCCC4CCOCC4)C3)=O)CCCN(CCC1)C2 N1(C(c2cc(C)ns2)=O)CC2CC(NC(=O)CCC3(C)CC3)CC2C1 N1(C(c2ccc(SC)s2)=O)CCC2(C)CN(C(c3cc(Cl)cn3C)=O)CC12 O=S(=O)(c1ccnn1C1CC1)N1CC2ON=C(C3CC3)C2C1 S(=O)(=O)(CCC(=O)N1CC2CC1C2C(=O)NC1CN2CCCC1C2)NC CCCCC(C(=O)NCC(n1cc(-c2c(F)cc(Cl)cc2F)nn1)C)C(C)C CC(C)(C)C(C#N)C(=O)N1CCC12CN(C(C1CC(C)(F)C1)=O)C2 c1(C(N2CC(C)OCC2)C(=O)NCCON)cccc([N+](=O)[O-])c1 N1(C(CCc2cnn(C)n2)=O)CC(NC(=O)CN2CC(=O)NC2=O)CC2(CC2)C1 c1(C(=O)NCCCCN(C)C(c2ccco2)=O)ccsc1C(F)F.C1(=O)CCN1 N1(C(C2N(C(c3scc(OC)c3)=O)CC(O)C2)=O)CCS(=O)CC1C c1(C(N2C(CCNC(C(CC)CC)=O)CCCC2)=O)ccc(OC)c2occc12 C1(C(N2CCC(N(c3nc(NC(C)=O)cs3)CCO)CC2)=O)CCOC(C)(C)C1 Cc1ccc(C(N2CC3(CO)CC2(C(=O)NCCC2CCCC2)C3)=O)cc1CO Cc1csc(=NCC(=O)N2CC(C)(C)CCC2CNC(c2ccc(CO)o2)=O)[nH]1 C1(NC(Cc2nc(C)c(C)s2)=O)CCN(C(=O)Cc2ncn(C)c2C)C(C)C1 C1(NC(=O)Cc2cnc[nH]2)CCC2CC1CN2C(=O)CCn1cc[nH]c(=O)c1=O N1(C(C(ON=C(C)C)C)=O)CCOC(CC(=O)NCc2ccc(C)n2C)C1 N1(C(Cc2scc(C)c2)=O)CCOC2(CCCN(C(=O)CC(C)P(C)(C)=O)C2)C1 N1(C(c2ccc(CC)s2)=O)C(CNC(C2CCS(=O)(=O)N2)=O)CC2CC12 C1(OC)(CNC(c2cocc2C)=O)CCN(C(=O)CC(C2CC2)C2CC2)C1 CON1CCC(CC(=O)NCC2(O)CCN(C(=O)COC3CC=CC3)C2)CC1 c1(OC)ccc(C(F)F)cc1NC(=O)OC(C)(C)C.c12cc(no1)C(=O)NC2 N1(C(CC2CC(=C)C2)=O)CC2CCCC2(NC(=O)C=C(C)c2ccccc2F)C1 CC1CN(C(c2ccc(Cl)cc2N)=O)CCCN1C(C1CCCSC1)=O C#Cc1cc(C(N2CC3(CC3)CC2C(=O)NC(C)COCC)=O)ccc1C N1(C(c2ccc(Cl)cc2Cl)C(=O)NC)CCC2C(=O)NCC2C1 c12ccccc1-n1cc(nn1)C2OC.c1(CC(=O)N(CC=C)C)nc(CC)no1 C1(S(N)(=O)=O)(C(=O)NCCC2(O)CCN(C(C3CC(C(C)C)C3)=O)C2)CCC1 c1(C(=O)Nc2c(C(C)=O)cnn2C)c[nH]c2c(C(F)(F)F)cccc12 c1(COC)ccc(NC(=O)CSc2cnn(C(C)C)c2)cc1 C1(CNC(C2(OC)CCC2)=O)CC2(CCN(C(=O)CC3OCCC3C)CC2)C1 CC(C)CC(F)(F)C(=O)NC1CCN(C(c2nnc(O)cc2O)=O)C1C CC(CCC(=O)N1CCC(C(=O)N(C2CC3CCC2O3)C)CC1)N(C)C c1(C(=O)NC2(CCNC(CCC(C)OCC)=O)CC2)cccc2c[nH]nc12 c1(C(N(C2CCN(C(C(C)OCC=C)=O)C2)CC)=O)onc(C)c1C C(=O)(C(C)(C)C(F)(F)F)N1CC(CC(=O)NC(CSCC)C)OCC1 C1(CNC(CC(c2scc(C)c2)O)=O)CN(C(c2cc(CO)[nH]n2)=O)CCO1 c12ccccc1S2.C(C(O)CCNC(=O)C(C1CCOCC1)F)NC(CSC)=O CN1N=CC(C(=O)NC2CC(F)(CNC(=O)C(c3ccc(F)cc3)=O)C2)C1=O C1(CC(=O)Oc2ccc(OC(=O)OC(C)(C)C)cc2)CCCC2(CCC2)O1 C1(NC(CCC(NN(C)C)=O)=O)CN(C(C2COCC2(C)C)=O)CC2(CCC2)C1 CC(CN=c1nc2c(Br)csc2c(Cl)[nH]1)(C1CC1)NC(c1ccn(CC(F)F)n1)=O C1(C(=O)NC(CCOC)C(N)=O)CC12CCN(C(=O)C(CC(C)C)N(C)C)CC2 c1(OC)ncnc(N2CCC(O)(C(=O)Nc3ccc(SC(C)(C)C)cc3)C2)c1C C(C(C)(C)C#N)NC(=O)CSSC.CC c1(C(N2C(C(=O)Nc3cccc(SC)c3)CC(O)C2)=O)cccn2cncc12 Cc1c(CCC(=O)NCCCC(C)NC(C2(F)CC=CCC2)=O)cnn1C c1(COC)ccnc(C(=O)NCC2(F)CC(NC(=O)Cc3ccns3)C2)c1 C1(C)(CNC(C2C(C)=CCS2)=O)CCCN(C(=O)Cc2nn(C)cc2Cl)C1 Cc1cn2ccnc(C(N3CC(CNC(=O)COCCO)CC3C)=O)c2n1 C1(NC(C(Cn2cncn2)NC(=O)CN2CCSCC2)=O)CC2CC3C(C2)C13 C1(C(N2CC3C(CNC(C(C)(C)C(N)=O)=O)C3C2)=O)Cc2n[nH]cc2C(=O)N1 C1(NC(Cc2scc(C)n2)=O)CCN(C(C2CCCCN2C)=O)CC1C c1(CC)cc(C(=O)NC2(C)CN(C(c3cccc(Cl)c3)=O)C2)n(C)n1 c1(OC)nn(C)c(Br)c1C(=O)NCCC(C)NC(=O)Cc1csc(=N)[nH]1 c1(C(N2C(CNC(=O)C(c3ccc(F)cc3)CO)CCC2)=O)cc(Cl)ccc1F C1(O)(CN(C(=O)CNC(=O)C2CC2)C)CCCN(C(=O)Cc2ccccc2)C1 c1(C(=O)OC)ccc(CNC2CCCC(C(=O)NC3(CO)CC3)C2)c(C)c1 CCCCCCCCN(S(=O)(=O)c1cccs1)C(=O)NC(C)CCCCO Cc1nc2c(s1)CN(C(C1(C)CC(NC(C3COC(=O)N3)=O)C1)=O)C2 n1(CC)nc(C(=O)NC(C2CC(NC(C3(CC4CC4)CCC3)=O)C2)C)c(C)n1 CCC(CC(=O)NC1(C)CN(C(c2ccn(C)c2C2CCC2)=O)C1)C(C)C C=C(C)C1OCCC1C(N1CC2(CC2)CC1C(N1CCC(C)(O)CC1)=O)=O N1(C(CCN(C(C)=O)C(c2ccc(C#N)s2)C2CC2)=O)CCCC2CCCCC12 c1(CNc2ccc(C(=O)N(CC(N)=O)CC)o2)ccsc1CC C#Cc1ccc(C(=O)NCC(C)NC(c2nn(C)cc2Cl)=O)c(OC)c1 c1(NC(CC(CC)CCc2ccccc2)=O)ccc(F)cc1F.C1(=O)CO1 N1(C(C(C)OCC#C)=O)CC2(C1)CN(C(=O)C(c1ccc(Cl)cc1)CO)C2 C=C=CCCC(=O)N1CCCC1N1CCN(C(C2C3CCC2CC3)=O)CC1 Cc1ccc2c(c1)CCCN2CC(=O)Cc1ccc(S(C)(=O)=O)cc1 C(=O)(CCS(C)(=O)=O)NCC(CC(=O)NC1COC(=O)C1)OC c1(C(C(C)NC(=O)CC2(O)CCOC2)=O)ccc(F)cc1Cl CC(C)C(C(=O)N(C)CCNC(c1ncoc1C1CC1)=O)n1cc(Br)cn1 C(CN=c1cc(NCC2(CO)CCC2)nc(C(C)C)[nH]1)(c1ccnn1C)OC c1(C(N2C(C(CNC(CC(C)C(F)F)=O)(C)C)CCC2)=O)ccc(C#N)c(F)c1 CCS(=O)(=O)CC(=O)Nc1cccc(C(=O)Nc2cnc(Cl)cc2C(N)=O)c1 N1(C(c2n(COC)ncc2)=O)CCCC(N(C)C(C2CC(CCO)C2)=O)C1 N1(C(c2ccc(N(C)C)nn2)=O)CCC(NC(=O)C2=CCC2)C(CO)C1 C1(C2C(NC(C=C(C)Cl)=O)CCO2)CCN(C(C2CC(CCO)C2)=O)CC1 C1(CNC(=O)CCC2CCCC2)CCCC(NC(c2[nH]nnc2C2CC2)=O)C1 c1(OC)c(F)cc(CNC(C2CCN2C(c2cccc(F)c2C)=O)=O)cc1F c1(OC)cccc(C(N2CCN(C(c3coc(C)c3)=O)C(C)C2)=O)c1N c1(C(=O)NC(C2CCCCC2)C(=O)N(CCC#C)CCO)cn(CCO)nn1 C#Cc1cccc(C(N2CC3CC2CC3NC(c2cscc2Br)=O)=O)c1 C(CCN=c1[nH]c(Cl)nc2c1S(=N)(=O)CCC2)NCCCC[Si](C)(C)C Cc1cc(C(=O)N(C(C)CNC(=O)C=C2CCC(C)C2)C)c(N)cc1F C1(O)(CNC(=O)CCn2ccnn2)CN(C(=O)NCC2CC2c2ccco2)C1 C1(C(=O)NCC2CCN(C(C(CC)C)=O)C23CC3)CN2CCCN1CC2 C1(CNC(C2CN(C(C(=O)NCCOC)=O)CC2C)=O)CCc2ccccc2O1 C1(NC(CC2(C#N)CC2)=O)CCCN(C(=O)CC23CCC(CC2)C3)CC1 C#CCCN=C(NCC1CC12CC2)N(C)Cc1ccc(OC)cc1F Cn1cc(C=CC(=O)N(C2CN(C(=O)Cc3ccccc3)C2)C2CC2)cn1 N1(C(c2cc(CC)on2)C(=O)NCCC(=O)OCC)CC(C)(C)OCC1C(N)=O c1(OC)ccc(C(=O)NC2CC2NC(=O)CC2CC3CC3C2)c(OC)c1 C1(NC(C=CCC)=O)CC(F)CN(C(=O)C(C)(C)C2CCOCC2)C1 Cc1ccn(CC(=O)NCC2CCCN(C(=O)C(C)(C)CF)CC2)c(=O)c1 c1(CN2CCCC(CC(=O)Nc3ncc(OC)nc3)C2)cc([N+](=O)[O-])cs1 CC1(C)CC(NC(c2cc(Br)co2)=O)CN(C(=O)CNC(N2CCCC2)=O)C1 C1(C(N2CCC3(CC(NC(C(N)=O)=O)C3)C2)=O)CC(c2cccc(F)c2)=NO1 Cc1oc(C(=O)NC2CCN(C(=O)C(c3ccc(Br)cc3)C)CC2)cc1CO N1(C(=O)C(=O)NC2CC(Oc3ccccc3F)C2)CCC(CCN(C)CC)CC1 Cc1ccc(C)c(C(N2CC(CNC(c3cccc(F)c3N)=O)CCC2C)=O)n1 N(C(=NCC(=O)N(C)C)N(C)Cc1csc(C)n1)CC(COC)(C)O c1(C(N(C(CNC(C(F)=CCC)=O)C)C)=O)cc(C(F)(F)F)cs1 c1(NC(C2CC(=C)CN2C(C2CCCOC2)=O)=O)cc(Br)cc(C(=O)OC)c1C CCC(C)CCC(O)CC(=O)N(CC(CO)(CO)NC(=O)C=CBr)C C(C(CC(C)C)C(=O)N1CCC(COC)C1)NC(COC1(C#C)COC1)=O CC1(C)CCN(C(C2(c3cccs3)CC2)=O)CC1CNC(=O)C1=NNC(=O)CC1 c1(C(=O)NCC(CC)NC(c2cc(C(N)=O)cc(F)c2)=O)cccc2scnc12 C1(O)(CNC(C=CC)=O)CCN(C(c2cn3c(n2)SCC3)=O)C1 C1(NC(COC(CC)C)=O)CCN(C(C2(c3ccccc3C)CCCC2)=O)CC1F c1(C(=O)NC(C)C(=O)NCCC(=O)NC2CC2)cnc2c(c1)CNC2=O C(CC(=O)N1CC(N(C)C)C(C)C1)(C(F)(F)F)NC(C(C)NC(CC)(C)C)=O C=CC1(C(N2CCC(NC(c3cc(F)ccc3C3CC3)=O)C2)=O)CCOCC1 CCC(C)C(O)C(C)C(=O)NC1CCCCC1CC(=O)NC(C)(C)C(O)C(F)F c1(NC(=O)CNc2ncccn2)ccc(CNC(=O)COCC2CC2)cc1F N1(C(c2ccc(Br)c(F)c2)C(=O)NCCSC)CCc2cc(C(N)=O)ccc2C1 C1(CC(=O)NCC(C(C)(C)C)NC(c2cc(Cl)ns2)=O)CCCC2(CCC2)O1 O=S(=O)(c1cc(Cl)c(Br)cc1F)NC1CCN(S(=O)(=O)c2nccs2)CC1F C(C1=NOC2(CCC2)C1)NC(C1C(CC)CCN1C(=O)CSC1CC1)=O C1(NC(C2CCCO2)=O)CN(C(c2cc(Cl)ns2)=O)CC1n1ccnn1 CC(C)(CCNC(c1ccccc1)c1nnnn1C1CCOCC1)N1CCCC1 C1(NC(c2c[nH]ccc2=O)=O)CCCN(C(C2CC2C(F)F)=O)C1 N1(C(C(C)(C)ONC(C(C2CC2)OC)=O)=O)CCC2(CCO2)C1 c1(C(=O)NC)sc2cc(C)ccc2c1Cl.C1C(=O)NCCOCCCCN1C.CC Cc1cc(C)c(C(N2CC=CC(NC(=O)C=C3CCCC3)C2)=O)cn1 Cn1cc(C(F)=CC(=O)NCCC2COCCN2C(=O)CC2CCSC2)cn1 C(=O)(C#CC1CCOCC1)NC1C2(CCN(C(c3c(N)cc(Br)cn3)=O)CC2)C1 c1(OC)ccccc1CC(=O)NC(C)CCN(C(=O)C(C)(C)C1CCCO1)C c1(C(N2CC(CN(C(=O)C(F)CC3CC3)C)OCC2)=O)cc2ccsc2[nH]1 Cc1ncc(C(=O)NCCN(CC(=O)OC2CN(C(=O)C(C)C)C2)C)n1C N1(C(CCC)=O)CCCC(C2CCN(C(=O)CN3CSCC3=O)C2)C1 c1(N)cccc(N2CC(N)CC2=O)c1.C(=O)(C(=O)NC(C)CNC(=O)C1CC1)CC CN1CCC(CC(N2CCC(O)(CN(C)C(C34COC(C)(C3)C4)=O)C2)=O)C1=O C=CCCCCCCCC(=O)N1CC(C)CN(c2ncc(I)cn2)C(C)C1 c1(C(N2CCC(CSc3ccncc3Br)C2)=O)c(F)c(F)c(Br)c(F)c1F c1(N2CC(CNC(c3cccc([N+](=O)[O-])c3)=O)OCC2)ncc([N+](=O)[O-])cn1 CS(=O)(=O)C1CCCN(C(=O)CC(Cc2cccs2)NC(c2ccc(Br)nc2)=O)C1 c1(C(=O)NCC(c2cccc(C)n2)(C)C)cc2nc(C)cc(C)n2n1 C12(C(C(C)=O)OC(C3CCS(=O)(=O)C3)=O)CC3CC(CC(C3)C1)C2 C1(NC(C2(C)CC2(Cl)Cl)=O)CCC(NC(=O)CCc2ccc(F)nc2)CC1 C1(CCC)C(=O)NCCN1C(C1CCC(NC(=O)Cn2nccc2C)CC1)=O c1(C(N2C(CCNC(C(N3CC(C)C3)C)=O)CCC2)=O)c(Cl)cnn1C(C)C C1(O)(CC(=O)NCc2cc(C(C)C)on2)CCN(C(c2cc(Cl)c[nH]2)=O)C1 N1(C(CCC#N)=O)CCC(CCC2CCN(C(C34CC(O)C3C4)=O)CC2)CC1 C1(NC(C2(COC)CN(C(=O)C(c3ccccc3)C)C2)=O)CCC(O)CC1 C1(C(=O)NCC(CC=C)NC(=O)CSC)CCN(c2ccc(Cl)nn2)CC1 CC1CN(C(C2CCCS2)=O)CCN1C(c1cnn(C)c1Br)=O c1(C(=O)NC2C(NC(=O)Cc3cc(C4CC4)no3)CC2)ccc(F)cc1Cl C1(C(C)NC(c2ccn(CCC)n2)=O)CN(C(C2C=CC=CC=C2)=O)CCO1 c1(C(N2C3C(NC(c4c(C)noc4)=O)(CCC3)CC2)=O)c[nH]c2c(Cl)cccc12 CC(C)C(C(=O)NCC1CCCCN1C(C1CC2(CCC2)C1)=O)c1ccn(C)n1 Cc1nscc1C(=O)NCCOC(C)(C)CNC(c1c[nH]cc1C(C)(C)C)=O S(=O)(=O)(CC(F)(F)F)CCNC(C(=O)NC(=O)NCCC(C)(C)C)CC1(C)CC1 C1(CC=C)(C(=O)NCCN2CC=CC2)CCCN1C(=O)COCCCN(C)C C(c1ccsc1C(F)(F)F)=CC(N1CC(CC(C)NC(=O)C(F)C2CC2)C1)=O N1(C(C(C(C(C)C)OC)O)=O)CCC2(CCCN(C(C3CC(CF)C3)=O)C2)C1 c1(N2CC3C(N(C)C)C3C2)ccncc1S(=O)(=O)NCCC(F)(F)C(F)F Cc1ccc(O)cc1C(N1CC(CNC(=O)CC2CCC2)CC1C)=O c1(C(=O)NCC2N(C(CC(CC)(F)F)=O)CC(OC)C2)c[nH]c2ncnc(O)c12 c1(C(=O)NCC(CO)NC(C(c2cccnc2)OC)=O)ccc2c(c1)CC2 C#CCCCCC(=O)N1CC(C(C)NC(c2csc(C(F)F)c2)=O)C1 N12CCC(CC1)C2=O.C12(C)CCN(C1)NC2=O.c1(SCCCC)c(C)coc1C C#CCC(CO)NC(=O)C(F)CC1CN(C(C2(NC(C)=O)CCC2)=O)C1 CC1CC(NC(c2cc(F)cc(Br)c2)=O)CCN1Cc1cnn(C)c1Cl C1(C(=O)NCC(CO)NC(C(C)=C(C)C)=O)CCC2(CC2)C1 C1(C)(C)C(=O)N2CCC(C2)OCC(=O)N1.n1(CCCNC(C)C)ccnn1 C1(NC(CC2C(C)=NOC2=O)=O)CN(C(=O)C(C)C)CC12CCS(=O)(=O)CC2 CCCS(=O)(=O)CC(=O)N1CC2C(NC(c3c(OCC)ccc(Cl)c3C)=O)C2C1 CC(C)(C)SC.C1C(=O)NCCNCCOCCO1.C(CSC)N C(=O)(C1=CC2C=CC(C1)C2)NCCC1(O)CN(C(C2C(C=C)CC2)=O)C1 c1(-c2c(C(=O)Nc3cccc(Br)c3F)cc(OC)nc2)c(F)cc(C)cc1F CC1Cc2cc(Br)cnc2N(C(=O)CC2(C(=O)O)CCC2)C1 C1(NC(c2nn(CC)nc2C)=O)CCCCCN(C(=O)CCOC2CCOC2)C1 N1(C(CC=C=C)=O)CCC(C(=O)N(C)CC23CCC(CC2)C3)CC1CC C1(NC(=O)Cn2cncc2)C2CCCCC12.C1(=O)CCN1.C1(OCCO)CC1 N1(C(CC(COC)C)=O)CC2CN(C(c3csc(C)n3)=O)CC2C1 C(=O)(C1=CCC(C)CC1)NCC1(NC(c2c(COC)nn[nH]2)=O)CCCC1 C1(CC)CCC(C)CN1OC(C)=O.C1(C)(C)C=CC(=O)N1CCNS(C)(=O)=O c1(C(=O)NC2C(C(=O)OC)CC2)cc(CNC(C2CC(C)(C)C2)=O)nn1C c1(C(=O)NCC(CCOC)NC(CCCC#C)=O)cc2c(C)c(C)ccc2[nH]1 N1(C(CC(C)CN(C)C)=O)CC2(C1)OCC1(CO)CC2(NC(=O)C=CCO)C1 C1(CC(=O)NCc2cc(C)oc2)CC(NC(=O)C(C)(F)c2ccccc2)C1(C)C C(=O)(C(CO)C(C)(C)C)NCC1C2N(C(C=NOC)=O)C(CC2)C1 C=CCCCCCCNC(c1cc(F)ccc1Br)c1nnnn1C1CCCCC1 N1(C(C2(COC)CCCO2)=O)CC=C(C(=O)NCC(C)CC(C)C)CC1 CCC(CC(=O)N(CCCN(C(=O)C#CC1CCCO1)C)C)C(C)C c1(OC(c2ccc(C)cc2Cl)=O)ccc(N(C2CCNCCC2C)CC)cc1O C1(CNC(c2c(CC)cccn2)=O)CN(C(=O)CC(C)(C)COC(C)=O)CCC1C C1(NC(c2c(C)nsc2)=O)CC(F)(F)CC1NC(=O)Cn1ncccc1=O c1(CC)ncccc1C(=O)NC1(CO)CCN(C(=O)CCc2ncc(F)cn2)C1 CC(C)(CCCNC(=O)Cn1ncnn1)NC(=O)Cc1ccsn1 N1(C=O)CC2C3CCC(C3)C2C1.c1(N(CCC)C(=O)O)ccc(Cl)cc1 Cc1cc2c(C(N3CC(NC(c4cocn4)=O)CC34CCC4)=O)ccc(C)c2[nH]1 c1(C(N(CC(CNC(C2(COC)CCC2)=O)(C)C)C)=O)cccc(O)c1[N+](=O)[O-] c1(NCC23OCC(NC(CSCCCC)=O)(C2)C3)nc(Cl)nc2ncn(C)c12 CCCCC(F)C(=O)N1CC(NC(c2cnc(OC)nc2C)=O)C2(CC2)C1 N12CCOC(C1)CC(C1CC1)CC2=O.c1(CC(C)C)cn(C2CCC2)nn1 c1(C(N2C3C(NC(C(C)OCC#C)=O)CC(CC3)C2)=O)c(C)ccc2nsnc12 N1(c2c3ncn(C(CC)C(C)C)c3ncn2)CCc2c(ncn2C)C1C C1(CC(=O)NCC2(C(=O)NCCC3CCCCC3)CCCO2)CN2CCC1CC2 c1(CCC(=O)NC(C(C)NC(C2C(OCC)C2)=O)C(C)C)ccc(Cl)c(F)c1 c1(OC)cc(C(=O)NC2CC(C)CN(C(c3cc(C#N)on3)=O)C2)cc(C)n1 N1(C(Cc2c(C)noc2C)=O)CC(C)(CO)CO1 c1(CN2CC(CC(=O)Nc3n(C)ccn3)C2)nc(Cl)ccc1F c1(C(N(C(CCNC(C(CC)=CC)=O)C)C)=O)ccc(C)c(S(=O)(=O)NC)c1 C(=O)(C(O)C(C)(C)C)NC(c1cn(C)nn1)C(=O)NC(c1cccc(O)c1)C N1(C(Cn2cc(COCP(CC)(=O)CC)nn2)=O)CC2(CCC2(C)C)C1 C1(COC)(NC(C2CC=C(C)CC2)=O)CCN(C(=O)CC2CCN(C)C2=O)CC1 N1(C(C2N(CC)C(=O)CC2)=O)CCC(C2(NC(=O)C(C)N(C)C)CC2)C1 c1(-n2cc(CCNC(C3C(OC(C)=O)C3)=O)nn2)cc(Cl)ccc1C c1(NCC(=O)NC(C=CC(=O)NC(C(C)C)C2CCC2)C)ccc(F)c(O)c1 N1(C(CCSCC)=O)CCC(CN(C)C(C2CC(F)(CF)C2)=O)CC1 N1(C(Cc2cc(C)nn2C)=O)C2CCC1CN(C(=O)CC1CCCC(O)C1)CC2 Cc1cc(C(=O)N(C2CN(C(=O)CC3CC(C(=O)N(C)C)C3)C2)C)sc1Cl C#Cc1cn(C)nc1C(=O)NC1C2CC3C1C3C2C(=O)NOCCF c1(C(=O)NCC(CC(C)C)NC(CCC#C)=O)cc2cccc(Br)c2o1 N1(CCC(N2CC(C)(NC(C(C3CCOC3)OCC)=O)C2)=O)CCC(O)CC1 C(C(C(F)(F)F)N1CCN(C(c2ccsc2)=O)CC1)NC(c1c(OC)nsc1)=O c1(C(N(C2CCN(C(C3COC(=O)N3C)=O)CC2)CC)=O)cccc(C(C)C)c1 c1(C(N2CCC3(C(NC(=O)C=C4CCC4)C3)CC2)=O)cc([N+](=O)[O-])cc(Cl)c1Cl C(=O)(CCCCCC(=O)NCC1CC1NC(=O)C=CC1CCOCC1)OCC c1(OC)ccc(CC(=O)NC2CC(NC(C3COC(=O)N3)=O)C2)cc1OC C(C(CC)CC(F)(F)F)NC(C(n1cc(CN(C)S(N)(=O)=O)nn1)C)=O c1(CN2C(CN3CCCC(CC=C)C3)CCC2)c(C)nn(CC)c1C CC1(F)CCN(C(c2cn(CCNC(C3(O)CC3)=O)nn2)=O)CC1 C(CO)(CCCNC(C1CCC(O)CC1)=O)NC(CC1CC(C)(C)C1)=O C1(C)(C(N2CCN(C)C(=O)C2)=O)CN(C(C2CCC(C)(C)OC2)=O)C(C)(C)C1 N1(C(C(C)OC)=O)CCC2(CC1)CC(NC(c1cc3c[nH]nc3cc1C)=O)C2 c1(C(N2CCCC(N(C(C(C(C)C)CO)=O)C)C2)=O)ccc(F)c(F)c1F Cc1cc(C(N2C3CN(Cc4cnc(Br)c(F)c4)CC23)=O)c(C)cc1Br C1(COC)CC(O)C(O)CC1NC(=O)C(=O)NCc1cccn1Cc1ccsc1 C(C)(C(=O)NCC(C)C(=O)NCCCC1(O)CCC1)(C1(C)CC1)OC C=C(C)CCC(=O)NCCCCC1CN(C(=O)CC(C)C2CCCCC2)C1 c1(C(C)C)cncc(C(=O)NCC2CCCC2NC(C2CC2CN(C)C)=O)c1 N1(C(c2ccc(CC(=C)F)cc2)=O)CCC2(CCCN(C(=O)CSC(=N)N)C2)C1 C(CC1CC1)(C(=O)NCC1CC(C)(O)C1)NC(CSCC#C)=O C1(NC(C2N(CC)CCCC2)=O)CCN(C(=O)C(F)(F)C2CC2)CC1C c1(NC(C2C(C(=O)Nc3c(OC)ncc(I)c3)C2)=O)csc2ccncc12 C1(NC(c2cnc(OCC)s2)=O)CCC(C)(CNC(=O)CCCN(C)C)C1 Cc1noc(C)c1CC(=O)NCC1CCC(NC(=O)C=C(Cl)Cl)CC1 C1(CNC(CC2(C)CC2(F)Cl)=O)CCCCN1C(=O)Cn1cncn1 N1(C(C2C(C)OCC2)=O)CC=CC(C(=O)NCC2(CO)CCCCC2)C1 N1(C(Cc2c(C)nsc2)=O)CC(NC(=O)CCc2cccnc2)CC1(C)C c1(CC(=O)NCCCCNC(C23CC2COC32CCC2)=O)cccc2nsnc12 c1(CC)ncc(C(=O)NCCC23C(C2)n2cc(nn2)C(C)(C)NC3=O)s1.CC.OC C1(CC(=O)NC2C(C)CC2)C=CC(NC(=O)C(N2CCOC2=O)C)C1 C1(NC(=O)C=C(Cl)Cl)CCCC12CCN(C(=O)Cc1nc(F)c(F)cc1F)CC2 C1(CC(=O)NCc2ccc(Cl)o2)C2CCC(C2)N1C(c1cnn(C(F)F)c1)=O C1(NC(C2(CC=C)CC2)=O)CCCCC1NC(c1cnc(-c2cccnc2)s1)=O C(CCC(=O)NC1CC(C)(NC(=O)CCCC2CCC2)C1)(C(N)=O)NC(C)=O C1(C)(CNC(C2CC(OC)C2)=O)CCN(C(=O)C(C)N2CCC2)C1 N1(C(CC(COC)C)=O)CC(C2(NC(C3CC3CF)=O)CC2)C1 N1(C(c2cn(-c3cccnc3)nn2)=O)CCN(C(C2(F)CC=CC2)=O)CC(O)C1 N1(C(C(CC)C)=O)CCC(C=CC(=O)NC2CCCC(F)(F)C2)CC1 CC1OC2(C(=O)NCC3(O)CC(NC(=O)C(F)CC4CCC4)C3)CCC1CC2 c1(CC(=O)N(C2CCN(C(C3CC3CF)=O)C2)CC)nsc2ccccc12 N1(C(c2ccc(CCC)s2)=O)CCN(C(=O)Cc2n[nH]c(=N)s2)CC1CCO N1(C(CSCC#C)=O)CC2CCC(NC(=O)CCCCOC)CC2C1 C(C(C)C(=O)N1CCC1CNC(C1C(C(F)F)C1(C)C)=O)SC N1(C(C(N)=O)=O)CCC(NC(C23CC2C3)=O)CC1c1ccccc1 N1(C(c2cc(C)n(C)c2C)=O)Cc2ccccc2C1C(=O)N1CC2OCCC12 N1(C(c2cccc(C)c2Br)=O)CC2CCC1C(CNC(c1ncoc1C)=O)C2 c1(OC)cccc(CCC(=O)NCCOCCCNC(C2CCCOC2)=O)c1 C12(C(N3CC(O)(CNC(c4c(OC)cccn4)=O)C3)=O)CC(C)(C1)OC21CCC1 C(=O)(CC(C)NC(=O)C(c1ccoc1)NC(=O)C(C)Cn1ccnc1)OC C12(CNC(CC=C)=O)CN(C(c3ccc4ccnn4c3)=O)CC1CCO2 C(CO)(C(=O)NCc1cn(C2CCC2)nn1)NC(=O)C1CC1.C1CN(C2CCC2)C1 CC1C(NC(c2nccnc2N)=O)CCN1C(c1cc(C(C)(F)F)n[nH]1)=O C1(O)CCN(C(=O)CCc2csc(C)c2)CC1.C(C(=O)NC)OCCOCCOC N1(C(CCC2CCCCN(C(C(CCF)OC)=O)C2)=O)CCCC2OCCC12 C(=O)(CC(C(=O)N1CCC(NC(=O)C=C2CCC2)C(F)C1)c1ccccc1)OC c1(C(=O)OCC)sc(C(C)NC(=O)CN(C)Cc2ccccc2)nc1C c1(C(N2C(C)CCC(CNC(CC=C)=O)C2)=O)ccc2c(n1)COCC2 c1(CC(=O)NC(CNC(C2CC(F)(F)C2)=O)CO)ccc2n[nH]cc2c1 CC1(NC(c2ccncn2)=O)CCCCC1C(=O)NCCCN1CCC1 C1(C(N(CCC(=O)NC)C2CC2)=O)CC2CCC1N2C(=O)C(c1cccnc1)O c1(OC)nccc(N(C(C2CC(N)C2)=O)Cc2cccc(O)n2)n1 CC(CC(F)(F)F)(C(=O)Nc1ccc(Br)nc1F)c1cccc(F)c1 C(=O)(C(C)(O)CC(C)C)N1CCCC(CC(=O)NC2(COC)CNC2)C1 C(=O)(CCC(C)(C)NC(=O)C(C)CSC)NCC(NOC(CC)C)=O C(=O)(C(CCCC)NC(N)=O)NC1C(CNC(c2c(COC)nn(C)c2)=O)C1 C1(NC(C=CCC)=O)CC1C1CCCN(C(=O)CCCOc2cccc(F)c2)C1 N1(C(c2ccc(OCC)cc2)=O)CCN(C(C2(F)CCOC2)=O)CC1CO C1(NC(Cc2ccc(C)cc2C)=O)CCC2(CC1)CN(C(C1CCC1C)=O)C2 c1(C(=O)NCC2OCCN(C(C(=O)NCCC(N)=O)=O)C2)cnc2c(c1)CCC2 c1(C(=O)NC2(CO)CCN(C(C3C(CC)C3)=O)C2)ccc(C)c(C#N)c1 C(=O)(C#CC1CCOC1)NC(C)C(=O)NCCn1cc(CO)nn1 C1(C=O)CN(C(c2ccc(C3CC3)nc2)=O)CC(C)(C)C1.CCCCNCCO C1(CC)C(C(=O)NC(c2cncs2)C)CCN1C(=O)Cc1coc(C)n1 C(=O)(C1CCCn2c(Br)cnc21)OCc1onc(-c2[nH]c(C)c(OC)c2OC)n1 C=CC(C)C(C)C(=O)N(C1CCC(NC(C2(F)CC=CC2)=O)CC1)C c1(C(N2C(CNC(c3cc(C4CC4)ns3)=O)CC2)=O)cc(=O)cc[nH]1 N1(c2n(C)c(C(c3ccccc3)O)nn2)CCC2(CC1)CC2Br C1(C)(COCC)CN(CC(=O)NCOC)CCO1 c1(OCCN(CCN(C(c2ccc(C)c(Br)c2)=O)C)C)ccc2ccccc2c1 C12(NC(C3N(C)C(=O)NC3)=O)CCCN(C(c3coc(CO)c3)=O)CC1C2 N1(C(C2CC23CN(Cc2cc(Br)cc(Br)c2)C3)=O)C2COCC1CC(F)C2 C#Cc1cnc(NC2CN(C(=O)CN3CC(=O)NC3=O)CC2C)nc1 N#Cc1ccc(NC(C2CNCCN2Cc2cccc(C3CC3)c2)=O)cc1Br c1(C(=O)NCC2N(C(C(CCSC)OC)=O)CCC2)cc(C)cc(Cl)c1 C1(SCCC)CCN(C(=O)Cc2nc(Cc3cccs3)no2)CC1 CCC(CNC(C1CC12CCOCC2)=O)N=c1[nH]c2ncnc-2c(C(F)(F)F)[nH]1 c1(C(=O)NCC(=O)N(CCC(C)O)C)cc(O)cc(=O)o1 N#Cc1cc([N+](=O)[O-])cnc1NCCC(=O)OCCC12CC(CC(=O)O)(C1)CO2 C1(NC(c2cn(C)nc2)c2nnnn2CC2OCCO2)CCC=CCC1 Cc1cc(C)c2cc(C(=O)NCC3CCN3C(C3(C)CCNC(=O)C3)=O)[nH]c2c1 C1(CC(=O)NCCn2cccc2)C=CC(NC(C2CC2C(F)(F)F)=O)C1 C#Cc1ccc(CNC(=O)CC2(CNC(C34CCCC3C4(F)F)=O)CC2)cc1 C1(NC(C)=O)C2CCN(C(=O)Nc3ccccc3-c3ccncc3)CCC12 C1(NC(c2cc(CC)cc(F)c2)=O)CCC2CCN(C(c3[nH]ccc3C)=O)C1C2 CC1(C)CC(=O)C=C(c2ccc(C(=O)NCC34CCCN3CCC4)cn2)C1 C1(CNC(C2N(C(Cc3cn(CC)nn3)=O)CC(F)C2)=O)OC(=O)CC1(C)C N1(C(c2cc(CC)no2)=O)CCC(O)CC1C(=O)NC1CC12CCC2 c1(C(C(=O)NC2CCC2)N(C)CCF)c(Cl)cnn1C CC(C)CC(C(=O)NC1CC(n2ccnn2)C1)NC(=O)CC1CCOCC1 c1(OC)c(C(=O)NCC2CC(C)N(C(=O)C(F)=CCCF)C2)cccc1Cl N1(C(=O)OCC)CCCC1C(=O)NCC1CCC1NC(=O)CCCc1nccs1 N1(C(c2c(CC)cns2)=O)CCC2(CC1)CC2NC(=O)COC1CC1 c1(C(N2CCC(O)(CNC(c3cn(C)nc3Cl)=O)C2)=O)cccn2nccc12 C1(C)(C(=O)NCC2(C)CCN(C(CCC=CC(C)C)=O)C2)CCCCC1C CC(C)CC1CNC(=O)CCNC1=O.C1CC(=O)N1.C(N)(=O)NC1CC1 C1(C(=O)NCC=CBr)C2CC1N(C(=O)CCC1CCOC1)C2 c1(N2CC(CN(C(C(C)SCCCC)=O)C)C2)nc2ccccc2o1 c1(C(=O)NCCN(CCCCCC)C(=O)Cc2cncs2)c(Cl)n[nH]c1C1CC1 c1(C(=O)NC(CNC(C(C)OCCC=C)=O)(C)C2CC2)cnn(CC2CCC2)n1 N1(CC2C(c3cn(CC(C)C)nc3)C2)CCC2CC12C CCCCC(CC)C(=O)NC(C)(CC)CCNC(c1ccc(CC2CC2)s1)=O Cc1cc(C(=O)N(CC(C)(C)NC(c2cccc(OCCF)c2)=O)C)cn1C N1(C(C(C)OCC)=O)CCCN(C(c2cccc(CC)c2OC)=O)CC1 CN1CCCC(CC(=O)NCCc2ocnc2CNC(=O)Cc2cnoc2)C1 c1(CCC2(C(=O)NCC(C)CNC(=O)CP(C)(C)=O)CC2)cc(CO)cc(F)c1 N1(C(C(C(CC)(C)C)OC)=O)CCCC2(CCN(C(=O)C#CC3CCOCC3)C2)C1 N=c1nc(CNCCc2cn3c(n2)SCC3)c(Br)c(N)[nH]1 CCC(CN(C)C)C(=O)N1CCC(CC(=O)NC(C)CO)CC1 N1(C(C=COCC)=O)CCC2(CC1)CN(C(C1CCCC3(CC3)C1)=O)CC(C)O2 c1(C(=O)NCC2C(CNC(C)=O)C2)cocn1 c1(OCC(=O)NCC2(F)CC(NC(C3CSC3)=O)C2)ccc2c(c1)CCCC2 C(=O)(C(C)(C)C(C)(C)C)NC(CNC(Cn1c(N)cc(C)n1)=O)C(C)(C)C N1(C(C2CCN(CC(=O)O)CC2)=O)CCC2(CC1)CCN(c1nnc(O)s1)CC2 c1(SC)cc(N2CCN(C)CC2NC(=O)CN2CCc3sccc3C2)nc(C)n1 C1(CNC(C(C)OCCN(C)C)=O)CCCCN1C(=O)CC12COC(CF)(C1)C2 c1(C(=O)NC2CC(CNC(c3ccn(CCC)n3)=O)C2)nccc2c1CNC2=O c1(NC(C(CC2CCC2)NC(C2CC(C)(C)OCC2)=O)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NC(C(CC)CCO)C)ccc2ncccc2c1.c12cnc(s1)C2 CCC(C)(COC)C(=O)N(C)CCNC(=O)C(C)CF N1(C(Cc2c(C)n[nH]c2)=O)CCC(F)(CNC(=O)CN2CCCC2CO)C1 c1(C(=O)OC)cc(Cl)c(N2CCC3(NC(=O)C4=C(C)CCC4)CCCC23)nc1C c1(SC)cccc(C(=O)N(C)CC2CCCN(CC3=CC=CC=C(C(=O)O)S3)C2)c1 c1(OC)ccc(N)c(C(=O)NCCCCC(C)NC(=O)CCCn2cncn2)c1 N#Cc1cc(C(=O)NCC2CCCC2NC(c2coc(C3CC3)n2)=O)cc(F)c1 c1(C(N2C(CNC(CCCS(N)(=O)=O)=O)CC2)=O)ccc2nc(Cl)nn2c1 CC1CN(C(c2ccnc(CO)c2)=O)CC1(C)CNC(c1coc(Cl)n1)=O C(=O)(C(F)CNC(N)=O)NCC(C)CN(C(=O)CC1(N(C)C)CC1)C O=S(=O)(c1cccnc1NCCCCF)NCCC1CCc2ccccc21 c1(NC(=NCC(C=C)C)NC2CCCC2)nc2cc3c(cc2[nH]1)OCO3 N1(C(=O)OC(C)(C)C)CCN(C(C23CCC(C2)OC3C)=O)CCC1(C)C C1(NC(C2CCC(C)(C)O2)=O)CN(C(=O)CCOC2CCC2)Cc2ccnn2C1 N12CCC3(CC3C1)NC2=O.CN1CC2CC(C1)C2NC(C1CC2C=CC1C2)=O C(=O)(CC(C)(C)CC(=O)N1CC2C(NC(C34CCN(CC3)C4)=O)C2C1)OCC c1(C(N(C)CC2(C(N3CC(NC(C)=O)C3)=O)CC2)=O)sccc1Cl C(=O)(C#CC(C)(C)C)N1C(CNC(c2nccc(COC)c2)=O)C(C)CC1 N1(C(CCCNC(=O)NCC#C)=O)CCN(C(c2csc(C)n2)=O)C(C)C1 CN1CC(=O)N(CC(N2CCC(NC(C3(Cl)CC3(F)F)=O)C(F)C2)=O)C1=O C(=O)(CCS(C)=O)N(C1CCN(C(c2ccc(N(C)C)cc2)=O)CC1)CC C(=O)(C(O)CCC(C)C)N(C(C(=O)NCC(CC=C)(C)CO)C)CCC N1(CC)CCOC(C(=O)NC2(CO)CCN(C(c3cn[nH]c3)=O)C2)C1 c1(C(N2CC(NC(C(CC)(C)F)=O)C(O)C2)=O)cc(=O)c2ccccc2[nH]1 C#Cc1ccc(CC(=O)N(C2CC3CNC2C3)c2nc(C3CCCC3)ns2)cc1 C1(=O)CC(C)(C)N1.c1(C(=O)NCC2CC(CC)C2)cn(C)nc1COC N1(C(c2ccc(C#C)o2)=O)CCCC12CCN(C(C1CC(OC)C1)=O)CC2 c1(C(=O)NCC2(C)N(C(CCC(CC)OC)=O)CCC2)coc(S(N)(=O)=O)c1 N1(C(CC(=O)NCC#C)=O)CCC(NC(c2ccc(CO)cc2F)=O)C12CCC2 c1(C(C)C)ccc(F)c(C(=O)NCCC2CCN(C(C3CCC(=O)O3)=O)C2)c1 C1(F)(C(=O)NCCN(C2CC2)CC)CCN(C(=O)CC(C)F)CC1 Cc1ncc(C(=O)N(C)CC2CC(F)CN2C(C2COCCN2C)=O)n1C CN1CCN(C(C2CNC(=O)O2)=O)CC1C(=O)NCCN1CCC1 N12CCCCC13CC(C3)NC2=O.c1(OC(C2CC(OCC)C2)=O)ccccc1 N1(C(C(C)OC)=O)CC(CNC(c2c(C(C)C)cccc2C)=O)CC(C)C1 Cc1ncc(C(=O)NC2(C(=O)NCC(F)CO)CC2(C)C)cc1C#N Cn1ncc(Cl)c1C(=O)NCC1C2CN(C(=O)C(O)Cc3cnc[nH]3)CC12 C12(C(=O)NC)CCC(F)(CO1)C2.C(CSC)(C(=O)N(CCOCCO)CC1CC1)OC C1(NC(c2cncc(C)c2)=O)CC2CC1CN(C(c1ccc(CO)cc1F)=O)C2 c1(C(N2C(C(C)(C)C(N3CC4C(C3)C4(F)F)=O)CCC2)=O)cc2cccn2cn1 C1(OC)CN(C(c2cnn(-c3ccccc3)n2)=O)CCC1NC(C)=O S(=O)(=O)(c1ccc(C#N)c(NC2CC(OC)C2)c1)NCc1cnn(CC)c1C C1(COC)(CNC(=O)COCC2CCC2)CCN(C(C2(C)CCC(=O)N2)=O)CC1 Cc1nnc2c(NC(=O)Cn3c(CC(C)C)nc4ccccc34)cccn12 CC1CN(C(=O)C(O)CCN(C)C)CC1CC(N1CCC(NC(=O)C2CC2)C1)=O Cc1cc(N)cnc1C(=O)NC1CCC(C(N2CCCC2(C)CO)=O)C1 c1(C(N2CCC(N(C(c3ccnn3C(C)C)=O)CC)C2)=O)ccnnc1S C(=O)(CCCC(C)NC(C1CCN(C)C1)=O)N(CCN(C(C)=O)C)C N1(C(C(C2CCC(C)CC2)CC)=O)CCC(NC(=O)C=C(C)C)C(CO)CC1 N1(C(c2n(C)c(Cl)cn2)=O)CCN(C(=O)Cc2cc(F)ccc2F)CC(C)(C)C1 CC(C)S(=O)(=O)c1ccc(C(=O)N(CCC2(O)CCOCC2)C(C)C)cc1 C1(NCCS(=O)(=O)N(C)C)CCCOC1c1nccn1CO.C(C)(C)(C)OC=O C(=O)(CCC(N)=O)NC(COCCOC)C(=O)N(C)CC1C2CCCC12 c1(CN2CC(C#N)C(C(=O)Nc3c(Cl)cc(Cl)nc3Cl)C2)c[nH]c2nccc(Br)c12 N1(C(=O)C(=C2CCCCC2)F)CCC2C(CCCN2C(=O)Cc2ccns2)C1 CC1CN(C(C2COC2)=O)CCCN1C(c1cc2ccncc2s1)=O CCN=C(NCC(c1cccs1)N(C)C)NCC(CCC1CCC1)OC(C)(C)C N1(C(COCC(C)C)=O)C2CCC(C2)C1CNC(C1CC12CC(F)(F)C2)=O C(C1CCc2ccccc21)NC(C1CC1c1ccc(F)cc1)C N1(C(c2c(CCC)n[nH]c2)=O)CCCC(NC(=O)C(C)CC(N)=O)CC1 C1(CCC(=O)Nc2c(CCC)n[nH]c2)CCCCN1C(c1cc(CC)nn1C)=O N1(C(C(C)c2cccs2)=O)CC(NC(C2CCC(C)C2)=O)CC1C Cc1ncnc(C(N2CC(F)CC2CNC(=O)CCOC2CCCOC2)=O)c1C C1(N(c2cccc(C(F)(F)F)c2)C(N2CCCC(C#N)C2)=O)(CO)COC(C)(C)C1 c1(C(=O)NC(CC(C)NC(CC(=C=C)C)=O)C)cc2ccc(Cl)cc2c(=O)o1 S(=O)(=O)(c1ccc2nc(N3CCOC(C(F)(F)F)C3)ccc2c1)NCC(=C)Cl CC1=NNC(=O)C1CC(N1CC(CO)C(CCO)C1)=O c1(C(N2CCC(N(C(=O)CC3(C)CCCC3)C)C2)=O)cc2cccnn2c1 c1(C(N(C(C)CNC(=O)CC(=O)OC(C)(C)C)C)=O)cc(N)ccc1O c1(NC(=O)C(c2cccnc2Cl)N2CCC(O)(C3N=NC=C3Cl)C2)ccc(F)c(Cl)c1 c1(OC)ccc(OCc2cc3c(N4CCCCC4)[nH]cnc-3n2)cc1S(C)(=O)=O NC1CCN(Cc2cc(I)ccc2Br)CCN(CC2CCC2)C1 CN1CCN(C(C2CCCN(C(=O)CN3CCC(=O)CC3)CC2)=O)CCC1=O N1(C(C2N(C(CNC(c3cccc(Cl)c3)=O)=O)CCC2)=O)CCC(O)(C(F)F)C1 C1(O)(C(CNC(=O)NC(C2CCO2)C)C)COC1 CC1(C)CC(NC(C2CC(=O)N(O)C2)=O)CCN(C(C2(C)CCCC2)=O)C1 n1(CC(C)(C)C)ncc(C(N2CC3CCC2C3)=O)c1-c1ccc(Cl)cc1 N1(C(CCCOC(C)C)=O)CC2COCCC2(NC(=O)CC2CCCOC2)C1 N1(C(c2cnc(OC)nc2)=O)CCN(Cc2cc(O)cc(Br)c2)C2CC12 C(C(C)CC(=O)NCCC1(C(=O)NC2C(C)C2C)CCC1)OC c1(OC)cnc(C(=O)NC(C)(CNC(c2ccccc2)=O)CC(C)C)c(OC)n1 c1(C(=O)NC(CCN(C(C(F)OC)=O)C)C(C)(C)C)ccc2nc(C)sc2c1 CCCC(CCCNC(=O)CC1(C)CC=CC1)NC(c1conc1C)=O c1(OC)ccc(SCC(N2CCCCC2CN(C)C(c2nocc2Cl)=O)=O)cc1 C(=O)(CC1=NNC(=O)C1)NCC1CC(NC(c2c(C)[nH]nc2Cl)=O)C1(C)C c1(C(=O)Nc2cccc(NC(C(C)NC(N)=O)=O)c2)onc2ccccc12 C1(N(C(=O)CCN(C(=O)CCC2CCC2)CCCO)CCCO)C=CCCC1 N1(C(c2nccc(OC)c2)C(=O)NC(C)C)CCC2(CSC2)C1 c1(-c2c(C)cco2)nc(CSc2ccccc2)n(C2CCSC2)n1 c1(C(CC)(C)C)ncc(NC2(c3nnnn3CC(F)F)CCN(C3CC3)C2)cn1 c1(C(=O)NCC(C2CCC2)NC(=O)CC2=CCCCC2)c[nH]c2nc(Cl)ccc12 Cc1ncc(C=CC(=O)NCC2CCN(C(c3n[nH]c(C4CC4)n3)=O)C2)c(O)n1 c1(CNCO)cc(OC)ccc1C.C1(N)CC(CC(C(CN(C(=O)OC)C)=O)=O)C1 C1(NC(=O)CSC(F)(F)F)CC(O)(CNC(C2CC(N3CCCC3)C2)=O)C1 C(=O)(C1=NOC2COCC12)NC(=O)CN(N1C(CC(=O)NC)CC1)CC(C)C N1(C(CN2CCN(C)CC2)=O)CC(CNC(C2CC3(C2)CC(O)C3)=O)C2(CC2)C1 N1(C(C23C(C)OC(CO)(C2)C3)=O)CC2(CC(NC(C3(C)CCCCC3)=O)CO2)C1 c1(OC)cccc(F)c1C(N1CCC(O)(CNC(=O)C=C(C)c2ccco2)C1)=O N1(C(C23C(C)(C)C(CC2)C3)=O)CCCC2CN(C(c3cccc(CO)c3)=O)CC12 C(=O)(C1=NNC(=O)CC1)N1CCN(C(=O)N(Cc2c(C)ccc(F)c2)CCN)CC1 N1(C(C(CC)OC2CCCC2)=O)CCC(NC(c2c(Cl)csc2Cl)=O)CC1C C(C1CN(C(c2sccc2CO)=O)CC1C(=O)NCCCCC1CCCC1)=CC C(=O)(C1=Cc2cc(C)ccc2OC1)N1CC(CC)C(NC(=O)CN(C)C)CC1 C1(NC(C2C(OCC)C2C)=O)CC2CCC(C1)N2C(C1(CCOC)CC1)=O N1(C(=O)OC(C)(C)C)CC(CNC(=S)NCCF)CC12CCOCC2 c1(CCN(C2CCCN(CCF)C2)C(=O)CC2CC3CCC2C3)c(Cl)cccc1Cl Cc1cccc(CC(N2CCOC(CCNC(C34CCC3C4)=O)C2)=O)c1 C12(C(N(CC(C(C)C)OC)C)=O)CCOC(C)(C1)C2 N1(C(C(c2ccc(O)cc2)C)=O)CCOC2CN(C(c3nccs3)=O)CC12 c12ccc3ncn(c3c1)CCNC2.C1(C(=O)OCC)(N)CCCCC1.OC C=CCN(OC)C(=O)C1CCC(CNC(C2CC2(F)Cl)=O)O1 C1(C(=O)NC)CC(O)CN1C(=O)CC1CCC(NC(=O)C=Cc2cccnc2)C1 CN1C(=O)C(C(=O)NCC(CO)NC(C2(CC3CC3)CC2)=O)Cc2ccccc21 C1(OC)CC(C)CN(C(=O)CC(O)CNC(=O)CC2CCCC3CC23)C1 c1(C(N(CCCN(C(C(CC)N(C)C)=O)C)C)=O)nc[nH]c2ncnc1-2 C1(C(C)C)CN(c2ccccc2)CCN1CC(=O)CC1CC1 c1(NC(c2nnnn2CCC2(C)CC2)(C2CC(=C)C2)C)cccc(C(N)=O)c1F C1(Br)(C(=O)NCC(C)NC(Cc2ccc(OC)s2)=O)CC12CCC2 C1(C(=O)NC(CSC)C)(SC)CCN(C(C2C(NC(C)C)C2)=O)CC1 N1(C(CCc2cc(C)n[nH]2)=O)CCCN(C(=O)CCCn2ccnc2C)CC1 N1(C(C(CC)N(C)C)=O)CCCCC1CNC(=O)Cn1ccc(Br)n1 CN1CCC(=O)N(CC2CC3(C2)OCCO3)C1=O c1(CCC(N2CCC(Nc3nccc(OCC)n3)CC2)=O)cnc2n1CCOC2 N1(Cc2cccc(OC)c2O)CCC2(CN(C(C3(C)COC3)=O)C2)C1 C=CC1(C(=O)NCC23CCC(CO2)C3)CCN(C(C2CC=C(C)CC2)=O)C1 C12(CNC(CCCNC(C)=O)=O)CC(CO1)N(C(C1(N(C)C)CCCC1)=O)C2 C(=O)(CCCC(=O)NCC(CO)NC(C1CCCCC1C1CCCO1)=O)OC CC(C)(CO)C(CN1CCCOC(c2ccccc2)C1)c1ccccc1 CC1CCc2sc(C(=O)NC3(CNC(=O)CN4CCOCC4)CCCC3)cc2C1 C1(CC(=O)NC2(CN(C)C(c3ncccc3N)=O)CC2)CCCCCC1 c1(C(=O)NCC(C2CC2)NC(=O)C(F)=C2CCCC2)ccc(Br)s1 C(C)(C(=O)N1CCC(N(c2cc(C)nc(CC3CC3)n2)C)CC1)(C(C)C)OC N1(CCC(C2CC2(C)C(F)F)C)CCN(C(=O)CC2CN3CCN2CC3)CC1 c1(C(=O)NC(C(C)NC(Cc2cnc(C)s2)=O)C)nc2ccccc2cc1F C1(CNC(C2C(CC)C2)=O)CC(F)(CNC(c2oncc2C)=O)C1 C1(C(=O)NC23CCC(CC2)C3)CCCC2(CC2)C1.C12(CSC1)C(=O)N2 CON(CCC(=O)NC1CCOCC1C)C(=O)CC12CCCC1C2 S(=O)(=O)(c1c[nH]ccc1=NC1CC1C)N1CCCC(Cn2c(C)cc(C)n2)C1 c1(C2C(C(=O)NCCCC3(NC(C(CCC)OC)=O)CC3)C2)cccc(C#N)c1 C1(NC(C=NOC)=O)CN(C(c2ccc(Cl)cc2F)=O)CC1C1CC1 C(=O)(CCC(C)OC)N(CC(C1CCC1)NC(=O)COCCC(C)C)CCC c1(Nc2ccc(OCC)c(C)c2)cc(C)c(F)cc1C CCS(=O)CC(=O)N(C(C)CN(C)C(C1CC1C(F)F)=O)C c1(C(N2CC(CNC(c3ccc(CC)nc3)=O)OCC2)=O)ccc(C)c(CO)c1 N1(C(=O)C=CCF)CC(CNC(=O)C(=O)NC2CC2)C2(CCC2)C1 N=c1[nH][nH]c2ccc(C(N3CC4CN(Cc5ccnn5C(F)F)CC34)=O)cc12 C(=O)(C(C)(C)S(C)(=O)=O)Nc1c(C(N2CC(OC)C(OC)C2)=O)nc(C)nc1 C1(C)(C(c2nnnn2C2(C)CC2)(C)NCCCCOC)CCOCC1.C(N)(=O)O c1(C(N2CC(O)(CNC(C3CC(C)OCC3)=O)C2)=O)cc(O)nc(Cl)c1 C1(CNC(C2C(C)=C2)=O)CCCC2CN(C(c3ccc(=O)n(C)n3)=O)CC12 Cc1[nH]nc(C(=O)NCc2ccc(Cl)nc2)c1[N+](=O)[O-].c12nc(cn1C)NC2=O C1(C(=O)NCCCCNC(CCc2ncc(C)[nH]2)=O)CCCSC1C c1(NC(c2ncnn2-c2ccccc2)=O)c(F)cccc1F C1(CNC(c2cc(OC)nn2C)=O)C2CCCC1N(C(C1CC(C)(C)CO1)=O)C2 C1(NC(C(=O)NCCOC)=O)CC(C(=O)NCCC2CCCC2C)CC1O c1(OCCC)ccc(C(N2CC(ON)(CNC(=O)CC(C)O)C2)=O)c(OC)c1 N1(C(c2c(Br)cnc(C)n2)=O)CCC2C(CCN2C(=O)CN2C(=O)CNC2=O)C1 c1(NS(CCCC)(=O)=O)ccc(S(=O)(=O)Nc2ccc3nnnn3c2)cc1 CC1(C)CN(C(c2ccc(Cl)c(N)c2)=O)CC1NC(=O)CCNC(=O)C=CCl C1(C2(C)N=N2)CCN(C(C2(NC(C3CC(=O)C3(C)C)=O)CCOCC2)=O)CC1 Cn1cc(O)c(=O)cc1C(c1nnnn1-c1cncnc1)NCc1cscn1 C#CCC(C)(C)C(=O)N1CCOC(C(=O)NCCCC2(C)CC2)C1 C=C(C)CCC(c1nnnn1CC1CCOC1)NCC1CC1c1cnn(C)c1 N1(C(CNC(=O)Cc2cccc(F)n2)=O)CCC2SC(=O)C=C2C1 N1(C(CCS(=O)(=O)N(C)C)=O)CCC(CO)C(NC(C2(CF)CCOCC2)=O)C1 C1(NC(c2c(CC)scn2)=O)CCC(C)(CNC(c2ccc(C)cn2)=O)C1 C(CCCC(C)(C)NC(=O)C=Cc1ccncn1)NC(C1C(C)OCC1)=O C1(NC(C2C3(CN(C(C(C)Sc4ccccc4)=O)C3)C2)=O)CCc2n[nH]cc2C1 c1(C(=O)NC23CC(NC(c4c(C)noc4)=O)(C2)C3)ccc(C(C)(F)F)nc1 c1(CCC(=O)NC2C(NC(CCn3c(C)ncc3)=O)CC2)ccncc1Br c1(C(N(CCN(C(c2cn(CC)nn2)=O)C(C)C)C)=O)cn2ncccc2n1 N1(C(COCC)=O)CC2(CCC2NC(C2CC(=O)N(CCN(C)C)C2)=O)C1 Cc1cccc(S(=O)(=O)N2CCNC(C(N3CC4CCC(C3)O4)=O)C2)c1 c1(CC(=O)NCC(=O)Nc2c(OC)cc(C(N)=O)cc2)cccc(S(C)(=O)=O)c1 C1(C(N2C(CCNC(c3c(CC)scc3)=O)CCCC2)=O)CC(C(C)(C)C)=NO1 N#Cc1cncc(C(=O)NCCC(=O)NCC(F)CO)c1 c1(NC(=O)NCc2cccc(CN3CCC(F)CC3)c2)ccc(Cl)cc1 N1(C(C(C)CN(C)C)=O)CCC(NC(C2C3COCC23)=O)C12CCCC2 CCCC(CC)CC(=O)NCCCN(C(C1CCCOC1)=O)C(C)C N1(C(COC)=O)CCC2(CCN(C(=O)NCC(C)C)CC2)C1 C1(C(=O)O)(OCC)CCN(C(C2CC=CC(N=[N+]=[N-])C2)=O)CC1 c1(C(N(C(CCNC(CC(CC)CC)=O)C)C)=O)cnc2[nH]nc(O)c2c1 N1(C(=O)C2=CCCCC2)CCCC2(CCCN2C(=O)Cc2cn[nH]c2)C1 c1(NCCOCCN(C)C(c2ccc3c(c2)COC3)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2sccc2Cl)=O)CCCCC2(C1)CN(C(=O)C(c1ccc(F)cc1)F)C2 N1(C(C=CC=CC)=O)CCC2C(NC(=O)CC3CCCOCC3)C12 N1(C(c2cc(OCC)n[nH]2)=O)CCC(CNC(c2ccc(N)cc2)=O)C1(C)C c1(SC(C)NC(=O)C(C2CCCO2)C2(NC(=O)OC(C)(C)C)CCC2)ccncc1 c1(C(=O)NC(CNC(c2c(C)con2)=O)C)n[nH]c(C)c1O C1(C(N2C(CCC)COCC2)=O)(NC(c2ccc(F)s2)=O)CCC(C)(C)C1 c1(C(=O)OCC)c[nH]ccc1=NC1CCCCCN(C(c2cncc(C)c2)=O)C1 N1(C(C=CC(=Cc2cnc[nH]2)C)=O)CC(NC(c2sc(CO)nc2C)=O)C(C)C1 Cc1sc2ncc(C(N3CC(O)C(O)C3CNC(=O)CN3CC=CC3)=O)n2c1C N1(C(c2cncc(CC)c2)=O)CCC2(CCCC2NC(=O)C(CO)C(C)C)CC1 N1(C(=O)NC(c2ccc3ncsc3c2)C)CCC12CCOCC2 C(C(=O)NC1CC1C)(c1cccs1)NC(COC(C)=O)=O n1(C(C)C)ncc2c(NCC(=O)N(C)OC)nc(N(CCCOCC3CC3)C)nc12 c1(CNC(N2CCC(O)(C(C(=O)NC)(F)F)C2)=O)cc(Cl)cc(S(C)(=O)=O)n1 CCCC(C)C(=O)N(CC(=O)N(C1CCN(C2CC2)C1)C)CC(C)C C(=O)(C1=C(Cl)CCOC1)N1CC(C(C(N2CC(CO)C3(CC3)C2)=O)OC)C1 C1(N(C(COCCCC)=O)C)CN(C(C2(C)CCCOC2)=O)CC12CC2 N1(C(CCC=C)=O)CC2CCC2(NC(C2CCN(S(=O)(=O)CCC)CC2)=O)C1 C1(C(=O)NCC(C)NC(c2cccc3oc(O)nc23)=O)CCC(C2CCCO2)O1 N1(C(c2c(C)noc2N)=O)CC(CNC(=O)CCc2nccs2)OC2(CCC2)C1 C1(CNC(c2cc(CO)ccn2)=O)C(O)C(O)CN1C(C1CC=CCC1)=O c1(OC)cccc(-c2ccc(CN(C)CCC3CCC(=O)N3C)s2)c1 Cc1nn(CCO)cc1NC(c1csc(C(F)(F)F)c1)=O Cc1ccc(OCC(N2CC3CC3(NC(C3CCCC(C)(C)O3)=O)C2)=O)c(C)c1 CON1CC(C(=O)NCC2(O)CCCN(C(c3cncnc3C)=O)C2)CC1=O c1(C(=O)NC2CC3(CN(C(C(C)CF)=O)C3)C2)ccc(S(C)=O)cc1 Cn1cc(N)c(C(=O)NC2CN(C(=O)CSCC3CCCCO3)CC2O)n1 CC1CN(C(=O)CCC2CCCCN2C(=O)C(O)CCC#N)C12CCOCC2 C1(CC)CN(C(c2c(C)noc2C(F)F)=O)CCC1NC(=O)C(C)SC N1(C(C2C(OC)CC2)=O)CCC(CNC(c2cc(N)cnc2Cl)=O)C1(C)C C1(COC)(CNC(c2ccccc2O)=O)CCCN1C(=O)Cc1ccsc1 c1(C(C)C)ccc(C(=O)N(C)CCOCCOCCNC(C2CCCO2)=O)cc1 C1(NC(C(CN(CC)CC)F)=O)CC(C)CN(C(=O)Cn2ccc(=O)cc2C)C1 C1(F)(C(=O)NCC(CNC(C(C)=C(CC)C)=O)O)CS(=O)(=O)CC12CCC2 C(C)(CCC(=O)NC(C)(C)CNC(c1cn(CC(C)C)nc1C(F)F)=O)SC CCCC(CCNC(C1(NC(=O)CNc2ncccn2)CC1(C)C)=O)C1CC1 C1(N(C(=O)CCc2ccn(C)n2)C)CC2CCC(C1)N2C(c1cnc(S)[nH]1)=O C1(CNC(C(CCC)N(C)C)=O)CN(C(C2CN(CC(C)C)C2)=O)CCCO1 c1(C(=O)NCC2CC(CNC(C(C)CF)=O)C2)ccc(C(O)CF)cc1 C(N=c1[nH]c2ccc([N+](=O)[O-])cc2s1)C1CCC(NC(c2ccccn2)=O)C1 CC(C)CC(Cn1cc(C2(O)CCOC2)nn1)NC(C1(C)CS(=O)(=O)C1)=O C1(NC(c2cc(F)ccc2C2CC2)=O)CCN(C(c2cc[nH]n2)=O)CC1F C12(NC(NC(C=C)C)=S)CC(C(=O)OCC)(C1)C2(F)F c1(C(=O)NC2C(C)CN(C(c3n[nH]cc3C(F)(F)F)=O)C2)c(N)sc2c1CCC2 Cc1c(Br)cnn1CC(=O)NC(C)CCNC(c1cc(CO)ccn1)=O N1(N2CCC2NC(C2CC(=O)C2)=O)CCCC2(CCC(OC)C2)C1.CC(C)(C)OC=O N1(C(CC(CC)c2ccccc2)=O)CCC2(NC(c3cc[nH]n3)=O)CCCC12 C(=O)(C1OCC(C)c2ccccc21)NCC(C)(C)NC(c1c(CCC)nco1)=O C1(O)(CCn2cc(CCC(=O)OC)nn2)CCN(C(c2cc(Br)co2)=O)CC1 C(C(=O)N(C)CC1(C)CCCO1)(C(C)(C)C)NC(C(C)CO)=O c1(C(C(=O)NCC(CN(C)C(c2coc(O)n2)=O)O)(C)C)c(F)cccc1F C1(NC(c2cccc(C)c2)=O)CCCC12CN(C(c1ccc(C)c(CO)c1)=O)C2 C123C4C5C1C1C2C4C51C(=O)NC1CCC(C1)NC3=O.c1(COC)cccc(F)c1 c1(-n2cc(CC(C(=O)OC)NC(=O)C(C)n3cccn3)nn2)ccccc1Br C1(CNC(CCc2nnc(C)o2)=O)(NC(=O)Cn2ccc(C)n2)CCCCC1C Cc1cc(F)ccc1S(=O)(=O)N(C1CCN(C(c2ccc(I)nc2)=O)C1)C CC(C)CC(CNC(=O)COC(F)F)NC(C1CN(c2ncccn2)C1)=O CC1(C=CC(=O)NC2(CO)CCN(C(C34CCC(CO3)C4)=O)C2)CCOCC1 C1(C(=O)NC2CCN(C(c3c(CC)ocn3)=O)C2C)CCC(C2CC2)C1 Cc1cccc(C(N2CCN(S(=O)(=O)C(Cl)(Cl)Cl)C3CC23)=O)c1[N+](=O)[O-] C1(NC(C(Cn2cccn2)NC(Cc2c(C)nsc2)=O)=O)CC2CC1C(O)C2O c1(-c2c(OC)cnc(Cl)c2)ccc2nccc(C(=O)Nc3ncccc3Cl)c2c1 C1(C)(Cn2cc(CCCN(C(=O)CCOCCO)CC)nn2)CCCC1(F)F c1(N(C)C)cc(C(=O)NCC2CCC(NC(c3cc(C4CC4)no3)=O)C2)n(C)n1 C=C=C(C)CC(=O)N1CC(NC(=O)CC(C)CN(C)C)C(F)C1 n1(CCC(=O)NC2CC(CCNC(=O)CN3CCSCC3)C2)ccc(O)nc1=O N#Cc1ccc(O)c(C(N2CCC3(C2)CN(C(C2(F)CC2(Cl)Cl)=O)C3)=O)c1 C1(C(C)C)N(C(C)C(=O)NCc2ccccc2)CC12CCS(=O)(=O)CC2 c1(C(=O)NCC2(O)CC(CNC(c3cn(C(C)C)nc3)=O)C2)occ2c1CCOC2 Cc1ccc(NC(=O)C(=O)NC2CN(C(C3COC3)=O)C3CC23)cc1Br c1(C(N2C(C)CC(NC(C(C)(C)SC)=O)C2)=O)cc2ccccn2n1 c1(C(N(C)Cc2cn(C3CCCC3)nn2)=O)cc(F)c2[nH]nnc2c1 N1(C(C(CCCC)O)=O)CCN(C(=O)CC(C)C(C)(C)C)CC(O)C1 c1(C(=O)OC)sc(Cl)cc1S(=O)(=O)N(C(C)Cc1cccc(OC)c1)CCO N1(C(c2cn(C)nc2Br)=O)CCC2C(CCCN2C(=O)CCC(N)=O)C1 CCC(CC)C(C(=O)N1CCC(NC(C2CCN(C)C2=O)=O)C1C(C)C)OC N1(C(C2CN(C)C2)=O)CCOCC1CCNC(c1cccc(-n2cccn2)c1)=O CCCCC(O)C(=O)NC1(C)CN(C(c2cc(C(=O)OC)cc(Br)c2)=O)C1 C1(NC(c2c(C)occ2)=O)CCCCN(C(c2nn(C)cc2N)=O)CC1 CCCCC(C(=O)NCc1cn(C2CN(C(=O)CC(F)(F)F)C2)nn1)N(C)C.C(N)=O c1(C(N2CCC(C)(CNC(C3(CC#C)CC3)=O)C2)=O)cc(C(N)=O)cc(C)c1 C1(CNC(c2c(CC)nc(C)o2)=O)CCCN(C(=O)CCSC2CCCC2)CC1 C=Cc1cccc(-c2cnc(Cl)c(C(=O)Nc3nc(Cl)cnc3OC)c2)c1 CCC(CC)(CC)C(=O)N1CCC(O)(CN(C)C(C2(C)CC2(F)F)=O)C1 C1(CNC(c2c(SC)ccs2)=O)CCC(F)(CNC(C2CC2CC(C)C)=O)CC1 Cc1cc([N+](=O)[O-])cnc1C(=O)NCC(C1CCCN1C(=O)OC(C)(C)C)(C)O N1(CCC(=O)N(CCNC(C2CC2c2ccccc2)=O)CC)CCCC(NC)C1 c1(OC)cccc(F)c1C(N1CCC(CNC(C2(OC)CC2)=O)(OC)C1)=O c1(NC(c2c[nH]c3ccncc23)=O)nc2ccccc2n1C1CCNC1 n1(CC)cc(Br)c(C(N2CCC(F)(CNC(=O)CC3CCC3(C)C)C2)=O)n1 CP(C)(=O)c1ccc(C(N2CCC3(C2)CN(C(C2(C4CCC4)CC2)=O)C3)=O)cc1 c1(C(=O)NC(C)CCCCNC(=O)C=Cc2ccsc2)cccn2cnnc12 C1(NC(C(OCC)OCC)=O)CCCC(NC(c2cc(C)c(C(N)=O)o2)=O)C1 c1(C(=O)NCC2(COC)CN(C(C3CCC(C)O3)=O)C2)cc(Cl)cn1CC C(C(CNC(=O)Cc1cnnn1C)C(F)(F)F)NC(c1c(OC)nccc1)=O C1(CC(=O)NCCC2(O)CN(C(C3CCC4CC4C3)=O)C2)CCC(F)(F)CC1 N1(C(c2c(C)nco2)=O)CC(NC(=O)CCCCCN(C)C)C2(CC2)C1 C1(C)(CNC(C=CCN(C)CC)=O)CCCN(C(c2cnccc2C(F)(F)F)=O)C1 CC(C)C(C)N=c1[nH]c(=N)[nH]c(=NCCCc2ccsc2)[nH]1 C1(C(=O)NCC2(NC(C3C(C)C3)=O)CC2)CCC2C(=O)NCC(=O)N2C1 CN1C(=O)CC(C(N2CCC2CNC(c2c[nH]ccc2=N)=O)=O)C1c1ccnn1C c1(C(N(C(c2ccccc2)COC)C)=O)cccc(C2CCOCC2)c1 CCS(=O)(=O)CCCSc1nnc(-c2cc(C)oc2C)n1CC(N)=O C(=O)(CC(C)(C)NC(=O)C1=CCCC1)NCCC(C)(C)N(C)C C1(NC(=O)NCC2CCCC(Cn3cc(CO)nn3)C2)CCC(C2CCC2)CC1 N1(C(c2ccnc(OC)n2)=O)CC2=C(C1)CN(C(c1ccc(N(C)C)nc1)=O)C2 C=C(F)C1(CC(=O)NCC(C)NC(C2CSCCS2)=O)CCOCC1 O(NC(=O)C(n1cccn1)NC(=O)CC(C)COCC)CCCC=C C1(N(C(C(=O)NCCNCC)=O)C)CC2CCC(C1)N2C1CC1 c1(C(=O)NCC2(CN(C(C(CC)OC)=O)C)CC2)csc2nccn12 CC1(CCO)CCN(C(=O)CC(C)(C)NC(C2CCSC2)=O)C1 C1(NC(=O)Nc2cc(SC3(Cn4cncn4)CCOC3)ccn2)CCCC(O)C1 c1(OC)ccc(CSC2CCC2(N)C(N2CCCCC2)=O)cc1 C(N=c1[nH]cnc2[nH]ccc12)C1CCC(NC(C2(C)C(C)(C)C2(C)C)=O)C1 CCCS(=O)(=O)CC(=O)NCC12CCC(NC(c3csc(C)n3)=O)(CO1)C2 c1(C(=O)NC2CC(CCNC(CC3(C=C)CC3)=O)C2)c(Cl)csc1Cl N1(C(Cc2c(CC)n[nH]c2CC)=O)CCC(F)(CNC(C2(C(N)=O)CC2)=O)CC1 N1(C(C(CCOC)(C)C)=O)CCC2CCN(C(c3ccn(CO)c3C)=O)CC2C1 c1(NCCC(C=C)(C)C)[nH]c(=NCCNS(C)(=O)=O)nc2c1ncn2C(C)C c1(C(=O)OC)ccc2c(c1)CCN(C(c1ccccc1-n1cccc1)=O)CC2 Cc1nccnc1C(N1CCCC(CCNC(C23CC(C#N)(C2)C3)=O)C1)=O C12(C(=O)NCC(C)CNC(=O)CC3CSC3)CCCCC(=O)N1CCC2 N1(C(C(C)SCC)=O)CCN(C)C(CNC(c2oc(C(=O)OC)cc2C)=O)C1 C1(C(N(C(C#C)C)C2CC2)=O)CCN(S(C)(=O)=O)CC1 C(=O)(CC(F)(F)F)NC(C(=O)NCC1N(C(C2(CC)COC2)=O)CC1)C c1(CC)nc2ccc(Cl)cn2c1C(N1CC(NC(=O)C2=CCCCO2)C(O)C1)=O C1(NC(C(F)OC)=O)CN(C(c2coc(CC3CC3)n2)=O)C2CCCCC12 C=Cn1nncc1C(=O)NCC(N1CCN(C(=O)C(C)C2CCCO2)CC1)=O N1(C(COCCCC)=O)CC(CC(=O)NCCN2CC3CC3C2)C(C)C1 C(=O)(CC1COc2ccccc21)NC(C(C)NC(C(CC)(CC)CC)=O)C C1(n2ncc(N(C(c3[nH]cc(C)c3)=O)C(c3[nH]cnc3C)=O)c2)CCS(=O)(=O)C1 C1(CCNC(COCCC(C)C)=O)CCCCN1C(=O)CC1CC=CC1 C(=O)(CCCC(C)NC(=O)C(C)NC(N)=O)N(CCC(=O)NC)CC1CC1 c1(C(=O)NCC(N(C(CSCC#C)=O)C)C2CC2)cccc2c1OCCO2 c1(C(N2C(C)CC(CNC(c3c(C)ccs3)=O)C2)=O)ccc(C(C)C)nc1C C1(Cc2cn(CCC(=O)N(C)C)nn2)CCCN(C(c2c(Br)cnn2C)=O)CC1 c1(CNC(=O)C(F)C(F)(F)Cl)cnn2c1CN(C(=O)C(F)OC(F)(F)F)CC2 N1(C(c2c(C)cc(Br)cc2)=O)CCC(F)(F)C(NCc2ccn(C)n2)C1 C1(CNC(C2C(C)C2)=O)CCCC12CCN(C(C1(C(F)F)CC(F)(F)C1)=O)CC2 C(=O)(CCCCCCSC)NC1(COC)CN(C(=O)C(F)OC(C)=O)C1 c1(C(=O)NCC2(NC(Cc3cn(C)nc3)=O)CCC2)cc2sc(=O)n(C)c2s1 C1(C(=O)NCC2CN(CC(F)F)C2)CCC(F)(F)CC1.C12COCCN1C(=O)N2 CCC(C)CC(C)C=C(CN=c1cc(C)nc(NCc2ccncc2)[nH]1)CO C1(NC(c2nn(C)c(Br)c2)=O)CN(C(c2ccc(O)nc2)=O)C2(CCOC2)C1 S(=O)(=O)(c1cccc(Br)c1F)N1CCC(CN(C)C(c2ccc(Br)nc2)=O)C1 c1(C(N2C(CC(=O)NCCSCCC)CCC2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(c2cnc(C3CC3)nc2)C(=O)NC)CCCC2(CC1)CNC(=O)C2 CCCC(N=c1cccc(S(=O)(=O)NCC2CCSC2)[nH]1)c1ccco1 C1(C(N2CCC(C)(CNC(C=CCN(CC#C)C)=O)C2)=O)CC2(CCCC2)C1 c1(C(=O)OC)cc(=NC2CCCC(CNC(=O)CCNC(N)=O)C2)[nH]c(Cl)n1 c1(CC(N2CC(O)(CCNC(C3C(CC)OCCC3)=O)C2)=O)c(O)ncnc1O CC(CC(=O)NCC1CCN(C)C1)N(C)C(c1cocn1)=O c1(C(N2CCC=C(C(=O)NCC)C2)=O)cnn2c(OC)cccc12 O=C(CCC1=CCCCC1)NC1COCCN(C(C2CCCSC2)=O)C1 c1(C(N(C)CC2CCCN(C(=O)COCCF)C2)=O)cc(Cl)cc2ccncc12 N1(C(Cc2cccc(SC)c2)=O)CCCC(C)C1CNC(=O)Cc1ccsc1C N1(C(CCC(C)OCC)=O)CC2CN(CCO)CC2C1 C1(C(N(CCC(N2CC(O)(CO)C2)=O)CC#C)=O)CC(C2CC2)=NO1 Cc1cc(C(=O)NC(C2CCCN2C(c2c[nH]cc2Br)=O)C)cc(N)c1 c1(C(C(=O)N(C2CCN(CC34CC5CC3C4C5)C2)C)(C)C)cccc2ccccc12 N1(C(c2nc(C(C)C)oc2)=O)CC2CC1CN(C(=O)CC(C)(C)C(F)F)C2 N1(C(c2ccc(C(C)C)s2)=O)CC(C)CN(C(=O)C(C)CN(C)C)CC1C C(=O)(CCS(=O)(=O)Cc1ccccc1)N(C1CCCC1)CCNC(CC=CC)=O Cc1nn(C)cc1S(=O)(=O)NC1CN(Cc2c(Br)ccc(F)c2F)CC1F c12cccc(c1)C(=O)NC2CN(C)C.Cc1ccsc1SNC(c1cscc1C)=O C(CCC)(C(=O)NOCC(=O)OC)NC(C(C)=CCN(C)CC)=O c1(C(=O)NC2CC3(CC(C(N(CC(CCC)O)C)=O)C3)C2)ccc2ccoc2c1 c1(C(N)=O)cccc(NC(=O)C#CCNC(C2(C(N)=O)CC2)=O)c1 c1(CNC(=O)CCc2cc[nH]n2)ccc2c(c1)CN(C(=O)CC1CCC(=O)N1)C2 C1(CNC(C2C(=C)C2)=O)CC(NC(C2(SCC)CC2)=O)C1 c1(SCC(=O)N(CCCCC2CCCN(C(=O)C(Cl)=CCl)C2)C)ncc[nH]c1=O C(=O)(CCS(=O)(=O)C(F)(F)F)N(C1CCCN(C(c2cc(C)oc2C)=O)C1)CC N1(C(C2(CCOC)CC2)=O)CCC(C(C)(C)NC(C2CSCCS2)=O)C1 c12ccc(cc1)C(C)NC2C.c1(OC)ccccc1.C(C)(CO)SCN C(C)(C(=O)N(O)Cc1cn(CCOC2CCCC2)nn1)NC(C(COC)(F)F)=O C1(NC(C2(C#C)CC2)=O)CN(C(C2(N3CCOCC3)CCC2)=O)CC1C CCC(CNC(C1CCN(C(=O)Cc2c(C)noc2C)C1(C)C)=O)(CC)CC C(=O)(CC(C)CC(C)(C)C)N1CC(C=C)(CC(=O)NOCC(C)(O)C(C)C)C1 C1(c2n(CC=C)c(SCC(C)C(N3CCCCC3)=O)nn2)CCCCCCC1 c1(CC)cc(N2CC3C(NC(=O)CCc4nccn4C)C3C2)ncn1 N1(C(C(C=C)O)=O)CCCCC(CNC(c2cc(C)cc(C)n2)=O)C1 C1(CNC(CC=CC)=O)CCC2(CN(C(=O)CCc3cnn(C)c3)C2)O1 CC1CN(C(c2c[nH]c(=N)s2)=O)CC(C)N(C(c2c[nH]nc2OCC(F)F)=O)C1 n1(CC)ccc(C(=O)N(C2CCN(C(c3cnoc3CC(=O)OC)=O)C2)C)c1C Cc1ccc(C(=O)NCC(C)N(C(=O)C(c2ncccc2F)(F)F)C)cc1CO c1(NC2CCC(C(=O)Nc3c(C)noc3)C2)ncnc2n[nH]cc12 C1(N(C)C)CCC(C(N2CC(NC(c3c(C(F)F)cnn3C)=O)C2)=O)CC1 C1(CNC(C2N(C(CCC)=O)CCC2)=O)CCCN(C(C2CCCC2(C)C)=O)C1 C1(CC)CCN(C(=O)Cc2cncc(C)c2)C(C(=O)NCCN2CCCC2C)C1 c1(N(C(c2ccc(=O)n(C)n2)C(=O)NC2CCCC2)C)ccc2c(c1)CCC2 C1(F)(CNC(Cc2cc(C)sc2)=O)CCN(C(=O)C=Cc2cc[nH]c2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC(NC(c2nnc(O)cc2O)=O)C(C2CC2)C1 N1(C(c2c(CC)nc[nH]2)=O)CCC2CN(C(c3cncc(C)c3)=O)CC2C1 C1(NC(c2cccc(O)c2Br)=O)CC2(C1)CC(NC(C1CCCOCC1)=O)C2 C1(CC(N2CCC(O)(CN(C(c3c(C)onc3)=O)C)C2)=O)CC2CCC(C1)C2 c1(C(=O)NC2CCC(NC(c3cc(C)ncn3)=O)CC2)c[nH]c2cccc(Cl)c12 C1(Nn2c(C(CC(COCC)C)CC)nnn2)CCOCC12CCCCC2 O=NN1CCCCC1C(=O)NCC1CCC(F)(CNC(=O)COCC(F)F)CC1 C1C(=O)NNC1=O.c1(OCCN(C)C)ccc(-c2nn[nH]n2)cc1 C1(NC(C(CC)C(F)(F)F)=O)CN(C(=O)CCCCSC)CCC12CCC2 c1(SCC(=O)NC(C2N(C(C(C)C3CC3)=O)CCC2)C)ccc(Cl)cc1Cl C1(NC(C(C)(N(C(C(C)N(C)CCN(C)C)=O)C)C2CC2)=O)CCCC1(C)C C1(NC(CC2CCN(C)CC2)=O)CN(C(=O)C=CS(C)=O)CC(F)(F)C1 C1(CC)(CC)CC(NC(C2(C)COC(=O)OC2)=O)CN1C(=O)Cc1ccnn1C C=CC(C)CC(=O)NCC(c1ccc(OC)cc1)NC(=O)CNC(N)=O c1(C(=O)NCCN2CCN(C(C(CSC)O)=O)CC2)cnc2c(C)cnn2c1 c1(CC)cnc(C(N2CCCC2C(c2ccc(OC)cc2)c2ccccc2)=O)nc1 c1(C(C)NC(CCNC(C)=O)=O)ccc2c(c1)CN(C(=O)C(F)C1CCOC1)C2 c1(NC(=O)CN2CCCCC2C2CCCNC2)ccc2c(c1)CC(C(=O)O)O2 C1(CC(c2ccc(F)cc2)NC(Cn2c(C)nnn2)=O)Cc2ccccc2C1C c1(C(N2CCCC(N(C(CC=CC=C)=O)C)C2)=O)nc(N2CCCC2)nc(=N)[nH]1 Cc1ncnc(C(=O)N(CCN(C)C(C2CC3CCC(C2)C3)=O)C(C)C)c1C CC1CCN(CCCO)C1C(N1CCC(NC(C2C3CC4C(C3)C24)=O)CC1)=O N1(C(c2nc(C)c(C)s2)C(=O)NCCN2CCOCC2)CCC(O)CC1(C)C CC(C(=O)NC(c1ccccc1F)CNC(=O)Cn1nccn1)S(C)(=O)=O C1(CNC(CNS(N(C)C)(=O)=O)=O)CN(C(=O)CCC(N)=O)CCC12CCOC2 c1(C(=O)NC2CCCC(NC(C(CC)N(C)C)=O)C2)cc2c(nc1N)CCCC2 c1(OC)cc(C)c(NC(=O)CC2(NCCNC(=O)CC(=O)N(C)C)CC2)cc1Cl C(C1=CCN(C(C2(CNC(C3CC(OC)C3)=O)CC=CCC2)=O)CC1)OC C(C)(C)(CC(=O)NCCC1CC1C1CC1)N(C)C(C1CNC(=O)C1)=O C#Cc1ccc(C(N2CC3C(C2)N3C(c2cc(Br)ncc2Br)=O)=O)c(Cl)c1 c1(C(=O)NCC2C3(CCN(C(CC#N)=O)CC3)C2)cnc2c(c1)COCC2 CCCCC(C(=O)NC1CC(CNC(c2cn3ccsc3n2)=O)C(O)C1)N(C)C c1(CNC(C2(NC(C3N(C)CC(O)CC3)=O)CCSC2)=O)cn2ccccc2n1 C1(NC(=O)C=CC2CCCO2)(CO)CCN(C(c2csc(Cl)c2)=O)C1 Cc1noc2nc(C(N3CC4(CC4)CC3CNC(c3coc(O)n3)=O)=O)ccc12 C1(NC(C2CCC(C)(C)CC2)=O)CN(C(=O)C(N)=O)C2CCCCC12 c1(C(=O)NCc2c(CC)nco2)ccc(CNC(=O)CC2CC(O)C2(C)C)cc1 N#Cc1cccc(C(=O)NC2CN(c3ncncc3I)CC2C#N)c1F C1(CNC(CCSC)=O)CCN(C(C2CCCN(C(C)C)C2)=O)C1(C)C n1(C(CC)C)nnnc1C(c1cncn1C(C)C)NCCCCF C(C)(c1ccco1)=CC(=O)NC1(CNC(C2(C)CC(=C)C2)=O)CCOC1 c1(C(=O)NCCC(=O)NCCCOCC)snc(C)c1N c1(C(=O)NCC2CCC(NC(c3cc[n+]([O-])cc3)=O)C2)cc2c(s1)CCCC2 Cn1ncc(CNC(C2(C)CC2(C)C)=O)c1C(=O)NCCc1c[nH]nc1O C1(CC(=O)N(CCOCCNC(c2ncc(OC)cn2)=O)C)OCCCC1(C)C c1(C(N2C(CNC(C(C=C)(C)C)=O)CC(F)C2)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 Cn1cnc(N2CCCC2C2(NC(=O)CN3CCCC3)CC2)cc1=O c1(C(=O)NCC2N(C(C(=COCC)C#N)=O)CC2)c(OCCOC)cccc1F CC1CN(C(C2(CNC(=O)OC(C)(C)C)CC=CC2)=O)CC1CN N1(C(C(CN(C)C)NC(CN(C)C)=O)=O)CC2C(CO)C2C1 C1(COC)CCCOC1.C1(CC(=O)NCc2ccsc2)CC(C2C(=O)N2C2CC2)C1 N1(C(C(C)=CC)=O)CCCN(C(=O)COCC2CCOCC2)C(C)C1 c1(OC)ccc2c(c1)C(C(=O)N(CCNC(=O)C(F)n1ccnc1)C(C)C)CCC2 C(C(CC1CC1)C(=O)N1CCCCC1C1(C)CC1)NC(c1ncn(CC)n1)=O N1(C(C(C)N(CC)CC)=O)CC(C)(C)CCC1CNC(c1cocn1)=O c1(OC)ccccc1CC(=O)NC(CO)C(C)NC(C1C2CCN1CC2)=O CC(c1ccccc1)=CC(=O)NCCCOCCNC(=O)CCCCNC(N)=O N1(CCC)CCCCC1C(=O)NC1CN(C(c2cccnn2)=O)CC1OC C(CN=c1nc2c(ncn2C)c(NC(c2cnsc2)C)[nH]1)NC(=O)NC C1(C)(CNC(C(C)O)=O)CN(C(c2ncn(C)n2)=O)C(C)(C)C1 c1(CCC=C)ccc(C(=O)NCc2cccc(CNC(c3cnco3)=O)c2)cc1 Cc1nn(CC(F)F)c(C)c1C(=O)N(C(C)C)CC1CCC1 C1(CC)C(C(=O)NCc2ccn(CC)n2)CCN1C(=O)CCNC(N)=O N1(C(c2cc(-c3ccccn3)[nH]n2)C(=O)NCCC)CCC(C)=C(F)C1 c1(N2CCN(C(=O)Nc3cc[nH]n3)CC2)nccc(=NCCC2CCCOC2)[nH]1 N1(C(c2c(C)oc(C(C)C)n2)=O)CCC(NC(=O)C(C)N2CCC2)CC1C n1(CCOC)c(C(=O)NCC(N2CCCC2)C2CCOC2)cc2ccccc12 C(=O)(CS(=O)(=O)CC(=O)N1CCc2sc(C3CCN(CC)CC3)cc2C1)OCC CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1CC1CNC(c1cnc(C(C)(C)C)s1)=O C(C(=O)N1CCSCC(C)C1)(C(C)(C)C)NC(CCCSC)=O CC1CCCN(C(c2cc(CO)[nH]n2)=O)C1CC(=O)NCC1(C2CCC2)CC1 N1(C(C(C)OCCC=C)=O)CCC(CN(C(=O)CSCC(F)(F)F)CC)C1 C1(NC(c2cccc(OC)c2)=O)CC2CC(NC(C3(C)CCCS3)=O)C2C1 N1(C(C=C(C)C)=O)CCN(CCN(C(=O)C(F)C2CCC2)C)CC1 c1(OC)ccc(-c2cn(CCOc3ccccc3Cl)nn2)cn1.C12CC1C(=O)NC2 C#Cc1ccc(C(=O)N(CC(=O)NCc2nccc(OCC)n2)C2CC2)cc1C CC(O)C(C(=O)NCCC(C)N(C)C(C1CC1(F)F)=O)N(C)C(=O)OC(C)(C)C C1(C(=O)NCC(C)CNC(c2ccc(-c3cccs3)cn2)=O)COC(C)(C)C1 S(=O)(=O)(c1ccc(S(=O)(=O)NC2CC(c3ccccn3)C2)nc1)N(C)C N1(C(c2n(CC)c(O)nc2)=O)CC(F)(F)CC1CNC(c1cc[n+]([O-])cc1)=O CC1CC=C(C(=O)NCC(CNC(C2(C)SCCCS2)=O)CO)CC1 C(=O)(C1=CCCN(C(=O)Cn2cccnc2=O)C1)NCC(C)(C)C#N C1(CC)C(C)CCN1C(C1CCN(C(=O)COc2cccnc2)C1)=O CC1CN(C(c2ccc(CN=[N+]=[N-])cc2)=O)CCC1NC(C1(C)CC1(F)Cl)=O C1(CCCCC)CN=C(NCC(C)C#N)N1.C(C)C C(=O)(C(CNC(=O)COCC1(O)CCCC1)N(C)C)N(C)Cc1nc[nH]n1 N1(C(N)=O)Cc2ccccc2C1C(=O)Nc1ccc(F)c(Cl)c1F N1(Cc2c(F)ccc(CC)c2)CC2CCN(C(=O)CCCCC(C)(C)C)C2C1 c1(NCc2c(C)cncc2)nc(N2CC3CCCCCC3C2)nc2c1ncn2C C(=O)(C(CC)C(C)C)NC1(C2N(C(CCCCC)=O)CCCC2)CC1 C1(NC(CCN(c2ccccc2)C)=O)CN(C(=O)Cn2cccc2)CCC1F c1(OC)cnc(Br)cc1C(N1CCC(O)(C(C)NC(=O)C(C)(C)CO)C1)=O CC(CC(=O)N(CCNC(c1ccccc1)=O)CCc1cnn(C)c1)C(F)F CC(CC(=O)NC(CNC(c1cc(N)ccc1F)=O)C(C)(C)C)C(F)F C=CCC(CC(=O)NCC1CC12CC2(F)F)NC(C1CCCC12CCC2)=O Cc1ccccc1Cc1noc(CCCCCc2cn[nH]c2)n1.N C(C)(C(C)CCCCC(=O)O)NC(c1cc(C)c(-n2cc(CO)nn2)cc1)=O N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC2(CCC(NC(=O)CN(C)C3CC3)C2)CC1 c1(C(N)=O)ccc(CC(=O)NCC2CCCN2C(=O)C(c2ccccc2)O)cc1 C1(CNC(C2C(=C)C2)=O)CCCN(C(c2ccc(-n3cccn3)cc2)=O)C1 Cc1nc(C(=O)NCC2CCC(F)(CNC(C3CC3F)=O)C2)nn1-c1nc[nH]n1 N1(CC(=O)NCC(CNC(c2[nH]ccc2C2CC2)=O)OC)CSCCSC1 c1(C(=O)NCC(C2CCCC2)NC(C2C(C)C2)=O)sccc1S(C)(=O)=O Cc1nn(C)c(C)c1CCC(=O)NC1CN(C(C2CCCCCC2)=O)CC1F C1(NC(c2ccc(Cn3ccnc3)o2)=O)COCCN(C(=O)C(O)CC(F)F)C1 C(N=c1[nH]cnc2c1SCCC2)C1CN(C(C(C)C(C)S(C)(=O)=O)=O)C1 N12CCCC(CC1)NC(=O)C2=O.C1(C(CC)NC(=O)CNC(=O)NC)CCCO1 COP(=O)(OC)C1CCCN1c1cc(=NCc2cc(C)co2)[nH]cn1 N1(C(CCC2(NC(C3CCN(C)C3)=O)CCC2)=O)CCCC(CCF)C1 N1(C(c2cncc(C)c2Cl)=O)CCC2(CCN(C(=O)CCc3cnco3)CC2)C1 N1(C(c2c(C)snc2)=O)CCN(C(C2CC2C2CC2)=O)CC1CF C(c1ccc(F)cc1)=CCC(=O)NCC1(CCNC(C(C=CCCC)O)=O)CC1 Cc1cc(C(=O)NC2CC(CN(C)C)CC2O)c(Br)c(Cl)c1 C1(C2CCN(C(C3CC(=O)N(CCC)C3)=O)C2)(NC(CCCCC)=O)CC1 c1(NC)cncc(C(N2CCOCC2CCC(=O)NC(C)Cn2cnnc2)=O)n1 C1(CNC(c2cc(C)c(C)s2)=O)CCN(C(=O)C2=CCCC2)CC1C CC1CC=C(C(=O)NCc2ccc(C(=O)OCC(F)(F)F)c(OC(F)F)c2)CC1 N1(C(CCCCOC)=O)CCC(C2CC(NC(c3sc(C)cc3Cl)=O)C2)C1 N1(C(c2c(C)nc(N(C)C)s2)=O)CCCC(CNC(c2nncs2)=O)CC1 c1(-n2cc(C(C)NC(C=Cc3cc(C)no3)=O)nn2)c(F)cccc1Cl C(=O)(CCCCC(=O)OCC)NC(CC)C(=O)N(C)Cc1ccoc1 Cc1nn(C)cc1CC(=O)NCCCNC(=O)CC1(C)CC1 Cc1cc(C(=O)OCCc2c(F)cc(Br)cc2F)nc2[nH]nc(O)c12 CC1CN(C(=O)NCC2N(C(=O)NC(C)(C)C)CCC2)CC1c1ccccc1 C1(CCOC)(NC(C2(CO)CCOCC2)=O)CCN(C(=O)CCCC(N)=O)CC1 c1(OC)ccc(CC(=O)NCC2(C)CCN(C(=O)CCCC#N)CC2)cc1OC C1(NC(c2cccs2)=O)CCC(O)CN(C(=O)C(c2cccc(Cl)c2)C2CC2)C1 c1(C(=O)NCC(C)(C)NC(=O)CC2CCCC23CC3)cc2c(Cl)cccc2[nH]1 CCC(C)C(C(=O)NCc1ncc(C)o1)N(C(=O)CC1CCCCCC1)C c1(CC)ccc(C(=O)NCC(C)(C(C)C)NC(C2CCC2C#N)=O)cc1 C1(CNCc2c(I)ocn2)CCCCC1C1CC1 C12(C(=O)NC3C(C)N(C(C4CCCC(C)C4)=O)CC3)CC3CC(C1)C(=O)C(C3)C2 N1(C(c2ccn(CC(C)C)n2)=O)CCC(NC(c2ccnc(CO)c2)=O)C(O)C1 C1(CC=C)(C(=O)NC2(CCCCO)CC2)CCCN1C(=O)CNC(C)=O C1(CC(=O)NCC(C)NC(=O)CCC2OCCO2)CCCOCC1 c1(CNC(c2c(CNC(Cc3cc(C)sc3)=O)c[nH]n2)=O)nn(C)c(=O)cc1C CC(C)C(CC1CCCC1)C(=O)NC1CN(C(c2cnsn2)=O)CC1C Cc1cc(OCC(=O)NC(C)CC(C)NC(=O)C(F)C(C)(F)F)cc(C)c1Cl n1(CC(C)NC(C=CC(C)NC(C2(OC)CC2)=O)=O)ccnc1 C1(NC(c2ncc(OC)nc2OC)=O)CCN(C(c2cocc2C)=O)CC1(C)C CC1(C)CC(C(=O)NCC2C(C)(C)C2(C)C)CN1C(=O)CCc1ncc[nH]1 c1(C(=O)NCCC(CCNC(c2occ(C)c2)=O)C)cc(F)cc(Br)c1O Cc1ccc(-c2cn(C3CN(C(C4(F)CCOC4C)=O)C3)nn2)cn1 CC(C)(C#N)CC(=O)N(CC(=O)NCc1ccc(C#N)cn1)C1CC1 c1(C(C)=O)ccccc1C(N1CCCC1Cn1cc(CC2CCCC2)nn1)=O c1(C(N2CCC(O)(CCNC(C3(OC)CCCCC3)=O)C2)=O)cc(C)cc(Cl)c1 C(CCC(=O)NCC(C)(C)CC1CN(C(C2CC(C)(O)C2)=O)C1)OCCOC C(C)(C(=O)NCC(CC(=O)Nc1c(C)noc1C)C1CCC1)(C(C)C)OC Cc1cc(C(=O)NC2(C)CCN(C(c3cc(N)ccc3C)=O)CC2)cc(C)n1 N1(C(CNC(C)=O)=O)CCCC1C1CCCN1C(=O)CSc1ncccn1 C1(C(CC)C)CCCCN1C(C1CC12CC(NC(C1C3CCC(F)C13)=O)C2)=O N1(C(c2ccc(C)c(C)c2)=O)CC(C)(C)OCC1CNC(C1CCC(=O)C1)=O CC1=C(C(=O)N2CCCC2(C)CC(N2CCC(C)(CCO)C2)=O)CC1 c1(C(=O)NC2(C)CN(C(C3CC(C(F)(F)F)C3)=O)C2)ccc2[nH]c(=N)sc2c1 N1(C(C(c2cscn2)N(C)C)=O)C2CCC1C(NC(c1cc(F)ccc1Cl)=O)C2 CCCC(CC)CCC(=O)N1CC(C(=O)Nc2c(C)cc(C)cc2C)C(C=CC)C1 C1(Nc2cc(NC(C)CS(N)(=O)=O)ncn2)CCOC2(CCOCC2)C1 N1(CCC#C)CCC(C(=O)NC(C)C(CO)NC(C2(CC#C)CCCC2)=O)CC1 N1(C(CCCc2onc(C)n2)=O)CC(NC(c2sccc2C(F)F)=O)C(C)(C)C1 C1(COC)(NC(=O)C(C)n2ccnn2)CCCN(C(C2CCC(C)O2)=O)C1 C1(C(=O)NCc2c[nH]nc2Br)CC12CCC(F)(F)CC2 CCCCC(C)(C)NC(=O)C(n1cc(C2(N3CCNC3=O)CCC2)nn1)C N1(C(c2c(OC)cccc2)=O)CCC2CN(C(=O)C(C)(C)CN(C)C)CCC2C1 c1(CN(C(C)C)C(=O)NC(c2cc(Br)no2)C)ccc(C(F)(F)F)cc1 CCC(CC)C(CCN=c1nc2scnc2c(N2CC(C)CC(C)(C)C2)[nH]1)OC Cc1ccc(F)c(C(N2CC3CC3(C(=O)Nc3c(C)nnn3C)C2)=O)c1 C(C)(C)(CCC(=O)NC(C(F)F)C(C)(C)C)NC(C(C)N1CCCC1)=O c1(C(N2CC3C(CNC(Cc4cc(C)sc4)=O)C3C2)=O)cc2cccnc2o1 N1(C(c2cc(C)c(C)s2)=O)CCCC2(CCN(C(C3CCC4CC4CC3)=O)C2)C1 Cc1cc(O)cc(C)c1C(N1CC(CCNC(c2cnsn2)=O)OC(C)C1)=O N1(C(C(=O)OC)=O)CCC2CCC(C1)N2CC1CCC(C(C)(C)C)CC1 C(N=c1ccc(S(=O)(=O)NCc2cccnc2CO)c[nH]1)c1c(C)onc1 c1(NC(C2CN(Cc3sccc3Cl)CCO2)=O)cccc2c([N+](=O)[O-])cccc12 c1(C2(C)CN(C(c3n[nH]cc3Cc3ccnc(F)c3)=O)C2)ccc(F)c(F)c1 Cc1nc(C)c(C(N2CC(NC(=O)CC3(C)CCCO3)CC(C)C2)=O)nc1C C1(C)(CC)C=C(C(=O)N(C2CC(NC(=O)C=CC(=O)OC(C)(C)C)C2)C)C1 C1(C)(CNC(c2n(CC)cnn2)=O)CC(F)(F)CN1C(C1CC(O)C1)=O Cc1nc(C)c(C(N2CCC(=CCNC(c3cccc[n+]3[O-])=O)CC2)=O)s1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CC(F)(CNC(C(C)N(C(C)=O)C)=O)C1 CC1=CCC(CCC(N2CC3CC2(c2cn(-c4ccc(C)cc4)nn2)C3)=O)CC1 C1(CNC(C(C)S(C)(=O)=O)=O)CCCC12CCN(C(C1(C)CC=CCC1)=O)CC2 C1(C(N)=O)CN(C(c2cccc(-n3ccnc3O)c2)=O)CCC1NC(=O)C(F)F C1(CNC(=O)C#CC2CCC2)CC12CCN(C(c1cscn1)=O)CC2 C1(NC(CCc2c(C)noc2Cl)=O)CC(O)CN(C(=O)CCc2ncccn2)C1 c1(CN2CCC(C(N(CCC(C)C)C)=O)C2)ccc(F)cn1 C(=O)(C(F)(F)CN=c1[nH]c(N2CCC(CF)C2)nc2c1COCC2)NCC CCC(CC)(CCC(=O)NCC(C1CCOC1)NC(=O)CCCOCC)[N+](=O)[O-] N1(C(C=CC(=O)OCC)=O)CCC2(NC(c3cc(C)ccc3Cl)=O)CC2C1 CCCC(C)(CC)C(=O)N1CC2CCC1C(CNC(=O)CC(C)C1CC1)C2 C12(NC(c3cn(CC)nn3)=O)CN(C(=O)CC3CCCCC3C)CC(F)(C1)C2 C=CCC(=O)NCCCN(CCO)C(C1CC(C(F)F)C1)=O N1(C(c2nc(OC)c(C)s2)=O)CCOC2(CCCN(C(c3sccc3C)=O)C2)C1 Cc1ccnc2c(C(N3CCC(CN(C)C(C4(C)CC(C)C4)=O)CC3)=O)cnn12 c1(CC)c[nH]c(C(=O)NC2(CNC(C3CC(C(C)C)C3)=O)CCC2)n1 N1(C(Cn2c(C)nnn2)=O)CC(O)C(O)C1CNC(C1(C)CC(C)(C)C1)=O N1(C(c2cccc(C)c2C)=O)CCC2CC1C(=O)N2 c1(C(=O)NCC2C(NC(c3cccc(CCO)c3)=O)CC2)cc2ccncc2s1 C12(CNC(C(C3CC3)OCC)=O)CCCC1N(C(c1csc(Cl)c1)=O)CC2 c1(C(N(C2CN(C(C(CC#C)C)=O)C2)C)=O)cc2cc(F)ccc2o1 OCC(CN=c1[nH]c(=NCCCOC(F)F)[nH]c2cc[nH]c12)c1ccccc1 C(=O)(CC(CC)C(C)C)N1CC(C(C)C)C(C(=O)NCCCOCCOC)C1 S1(=O)(=O)c2cccc(c2)N1.c1(OCCCOC)ccccc1C(=O)O Cc1cc2c(C(=O)Nc3ccc(NC(c4cncn4C)=O)cc3C)nccn2n1 c1(SCC(=O)NCC(C2CC2)NC(C2(C)CC(C)(C)C2)=O)ccsc1[N+](=O)[O-] CCCC(CC)C(=O)NC(CC(=O)NCC(O)CC(=O)OC)C1CC1 C1(NC(C(COC)N(C)C)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)C1(C)C N1(C(c2c(OC)c(C)cc(C)c2)C(=O)NC2CC2)CCc2[nH]nc(COC)c2C1 c1(C(N(C2CCN(C(=O)CC(F)(F)F)CC2)CC)=O)ccccc1F c1(CCC(=O)N(C(C)CNC(=O)CC(c2cncnc2)C)CC)cccc(F)c1 c1(C(N2CC(C)N(C(=O)Cc3cncnc3)CCC2)=O)cc(F)cc2nn[nH]c12 C1(NC(CCNC(=O)NC)=O)CCOCC1NC(C1(CO)CC(F)(F)C1)=O C1(C(=O)NCC2CC(CNC(C(OC)OC)=O)C2)(C(N)=O)CCCC1 N1(C(C(C(C)C)OC)=O)CC(CNC(C2CC3(C2)CC(F)(F)C3)=O)CC(C)(C)C1 C(=O)(C(CCOC)NC(=O)CCN1CCCC1=O)NCCC(C)N(CCC)C Cc1cccnc1CC(=O)NCC1CC(C(=O)NCCCP(C)(C)=O)CO1 CC1CC1C1CC1C(N1CCCC1Cn1cc(CNC(=O)Cn2ccnn2)nn1)=O c1(C(=O)NCCCCNC(CCC2N(C)CCCC2)=O)c(C#N)cnn1C N1(C(c2ccc(COC)cc2)C(=O)NCCC)CCN(C)CC1C C12(C(=O)Nc3ccc4cncn4c3)CCCC1CCN2CC(CC)C c1(C(N2CCCC(N(C)Cc3cc(Br)ccn3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(CCOC(C)=O)=O)CC2CC(NC(c3ccc(C(F)(F)F)c(C)c3)=O)CC1C2 N1(C(c2c(C)noc2N)=O)CC(NC(c2c(Cl)n[nH]c2C2CC2)=O)CC(F)C1 c1(C(C(=O)OC)NCc2cnc(-c3ccccc3)nc2)cc(F)cc(Br)c1 Cc1ccccc1CC(N1CC(CC(F)C(=O)NC2CC2C(N)=O)C1)=O N1(C(C(=O)NC(c2ccncc2F)c2ccccc2)=O)CCc2ccccc21 Cc1nc(C)c(C(=O)NC2(C)CCN(C(C3C(C(F)F)C3(C)C)=O)C2)[nH]1 c1(N2CCC(N(C(C(C)OCC)=O)C)C2)nc(C)nc(O)c1C c1(C(=O)NC(C)CC(=O)NCc2cccc(O)c2)nc(=N)cc[nH]1 C(=O)(C(C)C1CCCO1)NC1(CCNC(CSCCC)=O)CC1 C1(C(=O)NCC=CCC(=O)NC2C(C)(C)COC2)CC(=O)NC1(C)C C1(NC(C2(CCOC)CC2)=O)CCC(CNC(=O)CCc2ccnn2C)C1 C1(NC(=O)CC(c2ccc(O)cc2)C2CC2)COCCN(C(c2ccns2)=O)C1 Cc1ccc2cc(C(=O)NCC3CCCC3NC(C3CC(=O)N(C)C3)=O)cn2c1 C1(COC)(NC(=O)CCC2CCCCO2)CN(C(c2csnc2Cl)=O)C1 c1(C(N(C2CCN(C(CC(CCC)O)=O)C2)CCC)=O)cc2cc(Cl)ccc2o1 N1(C(c2c(OCC)n[nH]c2)=O)CCC2(CC1)CCN(C(=O)C(C)CN(C)C)C2 c1(C(=O)NC2CN(C(c3cn(CCC)nn3)=O)C(C)C2)cc(C)c2[nH]nnc2c1 c1(C(=O)OC(C)(C)C)ccc2nccn2c1.C1(C(=O)OC)CCN2C1C1(CC1)C2=O N(C(=NCCc1nccc(OC)n1)N(C)CC(C1CCC1)OC)C(C=C)C S(=O)(=O)(c1cccc2cccnc12)N1CCC(NC(C2(C)CCNC2=O)=O)C1 C(=O)(C1CCc2c[nH]nc21)NCC(CC)(CC)Nc1nnc(C)c(C)n1 c1(CCC(=O)NS(=O)(=O)CCCCl)cccc(O)n1.C123CC1CN(C2)C3 Cc1nc(C)n(CC(=O)NCC2CC(O)CN2C(=O)CN2CC(C)(C)C2)n1 CN=c1[nH]cc(C(=O)NC2(CCNC(=O)Cc3cc(SC)nn3C)CCC2)o1 N1(C(C(C(C)C)OC)=O)CCC(C)(C)C(NC(c2[nH]nnc2C)=O)C1 C(CO)(C(F)(F)F)NC(CNC(C1(NC(CN(C)C)=O)CC1(C)C)=O)=O Cc1ccc(N)cc1C(N1CC(O)(CNC(=O)COCc2nc[nH]n2)C1)=O c1(C(N(C(C(=O)NCC2C=CCOC2)C2CC2)C)=O)nn(C)cc1Cl C1(NC(=O)COc2ccccc2)CN(C(=O)CCCn2cccc2)CC1C1CC1 CC(C(=O)NC1CC1CCNCC(C)(C)OCC(=O)N(C)C)N1CCCC1 N1(C(c2ncn(CC)n2)=O)CCC(C)(CNC(=O)C(N2CCC(O)CC2)C)CC1 C1(CNC(c2cn(CCC)nc2)=O)C(C)CCN1C(=O)CNC(C)=O C#Cc1cc(C(=O)NC2CCC2NC(c2ccc(Cl)c(O)c2N)=O)cc(Br)c1 c1(C(N2CCC(C)(NC(C3CCC3(F)F)=O)C2)=O)cccc2nc(CO)[nH]c12 C1(CN(C(=O)CCc2ccsc2)CC)CCCN1C(=O)CCc1nc(C)no1 C1(CCC)CN(C(=O)C=CC(F)F)CC1NC(c1cnnn1C1CC1)=O N1(C(C(CC)n2cccn2)=O)CCN(C(c2c(C)noc2N)=O)CC(C)(F)C1 C(c1cc(C)cc(C)c1)=CC(=O)NC(CCCNC(CC1N(CC)CCC1)=O)C C1(NC(c2ccc(C(F)(F)F)cn2)=O)C2CC1N(C(C1CCOC1)=O)C2 C1(C(=O)NC2CN(C(c3cn(CC)nc3)=O)C2)C2CCC(C2)C1(C)C c1(C(N2CCC(N(C(=O)Cc3cnccc3Cl)C)CC2)=O)ccc(S(N)(=O)=O)s1 Cc1cc(S(=O)(=O)NC(C)C(C)C)ccc1-c1ccc2c[nH]nc2c1 CCC1=NOC(C(=O)NCC2CCN2CCc2n[nH]c(C)n2)C1.CN c1(C(=O)NC(CNC(C2OCCN(CC)C2)=O)C)cc(F)cc(Br)c1 C(c1ccccc1)(C(F)(F)F)=CC(N1CC(c2ccccc2)(CCO)C1)=O c1(CF)cc(F)cc2c1CCC2.c1(C2c3nnnn3CCON2)scnc1I N1(C(C=C(CC)C)=O)C2CCC1CC(CCNC(=O)CCn1ccc(C)n1)C2 CC(CN(C)C(c1ccc2ncnn2c1)=O)N=c1cc(C2CC2)nc(Cl)[nH]1 Cc1nc2cc(C(N3CCN(C(c4cnc(Cl)cc4Cl)=O)CC3CO)=O)[nH]c2s1 C1(C(N2CC(=C(CNC(=O)CCCc3ccccn3)F)C2)=O)CC2(CCC2)CO1 N1(C(c2sc3c(c2)CC(C)CC3)=O)CCOC2(C1)CN(C(C1CCCSC1)=O)C2 C1(C(=O)NC(CNC(c2cncc(C(=O)OC)c2)=O)C)CCc2ncncc2C1 c1(C(N2CCC(C)(CNC(=O)C=CCO)CC2)=O)cccc2[nH]nc(O)c12 C(CCCCCNC(C1CCOC1(C)C(C)C)=O)OCc1c(C(=O)OC)scc1 Cc1cc(Cl)c(C(N2CCC(C)C(N(C)C(C34CC(F)(C3)C4)=O)C2)=O)cn1 C1(CC(=O)NCC(CN(C)C(c2ncccc2O)=O)O)SC2=NCCN2C1=O CCCCC(C(=O)NC1CCC12CN(C(=O)Cc1nc([N+](=O)[O-])n[nH]1)C2)C(C)C C1(N2CCCC2)(CNCc2cncc(-c3ccc(C)cc3)c2)CCC2CCCC12 C=CCC(C(=O)NCC1(CNC(C2(C(=O)NC)CC2)=O)CC1(F)F)N(C)C c1(C=O)cnc2ccncc2c1.CCC(C(=O)N(CCOCCOC)CC)NCC c1(C(N2CC(N(C)C)C(CNC(=O)C(C)(C)F)C2)=O)nnn2c1CSCC2 C1(NCCCS(C)(=O)=O)CCN(C(=O)C(F)(F)Sc2ccc(F)cc2)CC1.CO C1(N(C(C2C(=C)CC2)=O)CC)CCN(C(c2csnc2-c2cccs2)=O)C1 O=C(CCCCC(F)(F)F)NCC(CC(F)(F)F)NC(C1CC2(CC2)C1)=O c1(C(N2CCC(C(N(CCCSC)C)=O)C23CC3)=O)cnn2ccc(Cl)c(F)c12 c1(CC)nn(C)cc1C(=O)N(CCNC(C1CCCNC1=O)=O)CCOC CC1CN(C(c2ccccc2)=O)CCC1C(N1CCC(O)(C(F)F)C1)=O c1(C(=O)NC2C(CNC(C(C)(C)OC)=O)C2)ccc(C(F)F)c(Cl)c1 C(=O)(N=c1cc[nH]c2ccsc12)N1CCN(S(C)(=O)=O)CC1 c1(NC(N2CCC(CC3CCCC(F)(F)CC3)CC2)=O)ncc(S(=O)(=O)C(F)F)cn1 N1(C(c2cccc(CC)n2)=O)CC(N=[N+]=[N-])CC1C(=O)NCCC1=CCCCCC1 CCC(C)C(C)C(=O)N(C)CCC1CCN(C(=O)CC2(N(C)C)COC2)CC1 C(CCC(C)(C)C(=O)N1CCC(C(N)=O)C1)NC(c1c(CC)cccc1)=O CC(C)(C(=O)N1CC(S(C)=O)C1)C1=CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 C(=O)(CC(=O)NC1(CC=C)CN(C(=O)CC(O)c2ccccc2)C1)NCC#C c1(C(=O)NC2CCN(C(CC(C)C)=O)C3C2C3)cccc(C2=CCOCC2)c1 N1(C(C(CC)(C)O)=O)C(C(=O)Nc2ccc(Cl)c(Cl)c2)C2CC(F)C1C2 S(=O)(=O)(c1cnn(-c2c(C)cc(C)cc2C)c1C)N1C(C(C(C)=O)O)CCCC1 c1(C(=O)NCCCCNC(CN(c2ccccc2)C)=O)cc2n(c1)CCC2 c1(OC)cc(CN2CCOCC2CC(=O)Nc2cncc(C3CC3)c2)c(Cl)cn1 N1(C(C(OC)OC)=O)CCN2CCN(C(=O)CN3CCCC3=O)CC2C1 CCCC(O)(CCC)CC(=O)N1CC2(CCN(C(c3nc(O)cs3)=O)C2)C1 N1(C(C2C(NC(CS(CC)(=O)=O)=O)C2(C)C)=O)CC2CC(OC)C(C2)C1 c1(C(=O)NC2(CN(C(C3OCCN(CC)C3)=O)C)CC2)n[nH]c2cccnc12 C1(C(N(CC(O)CNC(c2ccc(C#N)s2)=O)C)=O)CCn2cncc2C1 C(=O)(C1=CCN(C(C2CC23CCOCC3)=O)CC1)NCC1(C)COCCO1 C1(NC(C(C)(C)C2CC2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)CC1F C1(C(=O)NCC2(NC(c3cc(C)cc(N)c3)=O)CC2)CCC2COCCC2C1 C1(C(C)NC(=O)C(F)(F)c2cncs2)CN(C(=O)COCP(C)(C)=O)CCO1 c1(C(C)O)ccc(CN(C(Cn2cc(CC3CC3C)nn2)=O)C)cc1 C1(N(C(C=C(C)C(C)(C)C)=O)C)CCN(C(=O)CNc2ccccc2Cl)CC1C c1(CN(C(c2cc(CC)[nH]n2)C(=O)NC2CCOC2)C)cn2ccccc2n1 c1(NC2CCCCN(C(C(C)SC)=O)C2)nc(C)cc(C#N)n1 c1(C(=O)NCC(CNC(C(CC=C)C)=O)CO)cnc(O)cc1OC c1(CC(=O)NC2C(CNC(C3COCCO3)=O)CC2)ccc(F)c(F)c1 C1(CC(N2CCCC2C2(CO)CC2)=O)(OC)CN(C(=O)C(C)=CC(C)(C)C)C1 Cc1ccc(O)c(C(N2CCC(NC(c3sncc3Br)=O)C2)=O)c1 N1(C(=O)OC)Cc2cccc(NC(c3nnnn3C(C)C)C3COC3)c2CCC1 C(C#CCCO)NC(CN(C(=O)CC1CCC(=O)C1)CCOC)=O C(C(O)C(=O)N1CC=CC1C(=O)NCC1(n2nccn2)CC1)N(C)C C1(OC)(OC(C)(C)C)CC(O)C1.C1(CC(=O)O)CCN(C(=O)NC)C1 c1(C(=O)NC2C(C(=O)NCC3C(N(C)C)CCC3)COC2)cccc(F)c1F c1(OC)ccc(Br)cc1NCc1cnn(-c2ccccc2)n1 c1(CC(=O)NC(C2CCN(C(=O)CCn3cccc3)C2)C)ccncc1Cl C(=O)(C(CC(C)CC)NC(=O)C(C)C1(O)CCC1)NCC(NOCCOC)=O c1(C(=O)NC(CN(C(CC2CC(=C)C2)=O)C)(CO)CO)cc2ccccc2o1 N1(c2cncc(C(C)(C)C)n2)CCCC2CN(C(c3ccc[n+]([O-])c3)=O)CCC12 C1(CNC(CCN(C)C)(C)c2nnnn2C)CC2CN(C(=O)OC(C)(C)C)CC12 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCC2CC(O)CC(O)C2)C12CC2 C(=O)(C(C)(C)CCS(C)(=O)=O)NCC1(NC(Cc2ncn(C)c2)=O)CCCC1 c1(CC)ccc(-c2cn(CCN3CCN(C(=O)C(=O)NC(C)C)CC3)nn2)cc1 CC1CCC2(CCC2)CN1C(=O)C(N1CCN(C2CCCN(C)C2)CC1)=O C(=O)(C(C#N)C(C)(C)C)N(CC(=O)NCCC(CCC#C)O)CC#C C(CCCCNC(=O)COCc1ccccc1)NC(C=CC(=O)OCC)=O C(=O)(CCCCC)N(CCOCCCNC(CCC=CCC=C)=O)C C1(NC(=O)OC)(CC(C)CC(N2CCCOCC2)=O)CCOCC1 C1(OC)CC2CN(C(=O)C(F)C(C)CNC(c3cc(C4CC4)[nH]n3)=O)CC12 C1(CNC(CCCCC#C)=O)CCC2(CN(C(=O)CCC(C)SC)C2)O1 C1(C(N2CC(O)(C(C)(C)CNC(=O)CCSCC3CC=CC3)C2)=O)CCCCC1 C1(C(N2CCC(NC(c3ncc(OCC)nc3)=O)CC2)=O)CC2CCCCN2C1 C12(CC)CCCCN1C(=O)N(CCC1CCOC1)C2=O c1(NC(c2n(C=C)ncc2)=O)cc(F)ccc1NC(=O)NCCC N1(C(C2(OC)CCSC2)=O)CC2CCC(NC(=O)CSc3cccs3)(C2)C1 Cc1onc(-c2ccsc2)c1C(=O)NCC1CN(CC2COCCO2)CCO1 O=C(O)CCCS(=O)(=O)CCNCc1cc(F)ccc1I C1(c2cn(C(C)C(=O)N(CC(F)(F)F)CCO)nn2)CC2CCC1CC2 c1(C(C(=O)NC2CCN(C(c3cc(CCC)on3)=O)C2C)=O)cc(Cl)cc(Cl)c1 N1(C(c2n(CC)nnc2)=O)CC(NC(=O)CCCc2cccs2)C(C2CC2)C1 C(=O)(C1=C(F)CN(C(=O)C(C)n2cnnn2)CC1)N(C(C(C)O)C)C1CC1 N1(C(Cc2cc(C)nnc2O)=O)CCn2cnc(-c3ccccc3)c2C1 c1(CC)ccoc1C(=O)NCC(CCNC(=O)C(C)CC1CCC1)OC N1(C(C(C)CF)=O)CCN(C(c2ccc(F)c(CO)c2)=O)C(C(F)F)C1 C12(CC)COC(C(=O)NC3CCC3NC(c3ccc(CO)s3)=O)(C1)C2 C(=O)(CC1=Cc2ccccc2C1)NC(C1CN(C(C2CC(S(C)(=O)=O)C2)=O)C1)C N1(C(C(C)N(C(=O)Cc2ccnn2C)C)=O)CCCOC(C)(C)C1 C(CC(C(=O)N(C1CC(C)C1)C)NC(=O)C(C)c1ccsc1)SC C(=O)(CCC1=CCCCC1)NC(CC=C)CNC(=O)C(=O)N(C)C c1(C(N2CC=CC(NC(C=C(C)C)=O)C2)=O)cnc2sc(C)nc2c1 C1(C(=O)NC2CCCN(CC)C2)CC2(CC2)CN1C(=O)C#CC(C)C N1(C(CC2N(C)CCOC2)=O)CCOCC(C)(CNC(=O)C=Cc2nccs2)C1 CN1CCCC1C=CC(=O)NC1CC1NC(C1CC(n2cnnc2)C1)=O CCCCC(C(=O)NCCC(O)C(=O)NC1CC2(CC2)C1)C(C)C c1(NC(C2(CCNC(CCCC)=O)CC2)=O)cccc(NC(N)=O)c1 N1(C(C(CC)C(C)O)=O)CC2(C)CN(C(=O)Cc3ccc(F)cn3)CC2(C)C1 c1(C(=O)NC(CCC)C(=O)NCC(O)Cn2cccn2)ncc(C)cc1C N1(CCN(C)C(c2cnc(O)s2)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 C1(C(=O)NC2CC(CNC(c3c(CC)ocn3)=O)C2)(OC)CC(C)CC(C)C1 N1(C(=O)C=Cc2c(F)ccc(Cl)c2F)CC23CCCC2(COC3)C1 c1(C(C)NCC2(OC)CCCC2)ccc([N+](=O)[O-])cc1SCC C1(F)(CNC(CN(CCC(N2CCCC2C2C(C)C2)=O)C(N)=O)=O)CCCCC1 c1(OC)cc(C(=O)NCC(=O)N(C)C)ccc1NC(c1cnn(C)c1)=O C1(C(=O)NCc2ccc(C(C)=O)[nH]2)CN(C(=O)CC(C)(C)C)CC(C)(C)C1 C1(n2cccn2)(CNC(c2c(C)ccs2)=O)CCN(C(C2(C)CC2F)=O)CC1 Cc1cncc(CCC(=O)NCC(O)CNC(=O)C(C)(C)CN(C)C)c1 c1(C(N2CC(N(C)C(c3cc(C(F)(F)F)n[nH]3)=O)C2)=O)csc(N(C)C)n1 Cn1nccc1C(F)=CC(=O)Nc1cccc(-c2ccsc2)c1 C(CCCCC(=O)N(CC(N1CC(O)(CO)C1)=O)CC1CC1)=CC C1(COC)(NC(c2nc(C(F)(F)F)sc2C)=O)CCCN(C(=O)C2=CCC2)C1 N1(C(c2ncc(C)c(C)c2)=O)CCCN(C(c2occ3c2CCC3)=O)C(C)C1 c1(C(N(C2CC(NC(C(CC)OC)=O)C2)C)=O)cc(OC)c(Cl)cc1Cl C(Cc1ccco1)(C(=O)NC1(CO)CC1)NC(=O)CCc1cncs1 C1(NC(c2n[nH]c(C)c2F)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(C)C C1(CNC(CC2C(C)(C)C(N)C2)=O)CC2CNC1C2 Cc1nc2ncccc2cc1CCC(=O)NCC#CCNC(=O)C=CS(C)=O c1(C2CN(C(=O)NCCC3(OC)CCOC3)C2)nnc2n1CCC2 CC1CCN(C(C2CN(C3CCOC3)C2)=O)CC1NC(=O)CC1OCCC1C C(=O)(C1=CC2(CCOC2)C1)NC1C2(CCN(C(c3cc(CC)oc3C)=O)C2)C1 N1(C(Cc2nnc(C)s2)=O)CCC(NC(c2sc(C)c(C)c2C)=O)C(O)C1 c1(C(N(CC(=O)OCC)CC)=O)ccc(CNC(=O)C=Cc2scnc2C)cc1 c1(C(N(C(=O)CN2CCCC2CSC)CC)=O)ccccc1S(C)(=O)=O N1(C(Cc2ccc(C)cc2)=O)CC2CC1CN2C(C1(C2CCCO2)CCC1)=O CCCCC(CNC(=O)CC(C)(O)C1CC1)NC(C1CCC(C(=O)OC)CC1)=O C(CCCC(C)NC(c1sc(C)cc1OCC)=O)NC(CSCC=C)=O C(COC(C)(C)C)(C(=O)NCC1CCCN1CCCC=C)N(C)C C(CCC(C)C(=O)N1CCC(C)(CCNC(=O)COCC2CCOCC2)C1)OC c1(C(=O)NC2C(NC(C(C)Sc3nnnn3C3CC3)=O)C2)cnc2c(c1)COC2 N1(C(c2c(C)nsc2)=O)CC2(CC(C(=O)NCC3(C)CCCC(C)(C)C3)CO2)C1 CCCC(C(=O)N1CCC(C)N(C(c2cc(C#N)ccc2N)=O)CC1)C(C)C c1(C(=O)NCCC2CCCN(C(C3(C)CCNC3=O)=O)C2)nccc(Br)c1O CC1Cc2ccc(C(=O)N(C3CCC(C)(C)CC3)C)cc2O1 c1(C(=O)NCC2CC(F)CN2C(=O)CN2CC=CC2)cc2c(nn1)CCC2 c1(C(=O)NC(CC2CCOC2)C(=O)N2CCC2Cc2ccccc2)cc(Cl)cs1 Cc1cc(Br)cc(Cl)c1NC(=O)CC1CCC(NC(=O)CC2CCCC2)CC1 Cc1oc(C(=O)N(C)CC2CCCN(C(c3cccnn3)=O)C2)cc1S(C)(=O)=O c1(C(=O)NCC(C)(CNC(=O)CSc2nncs2)OC)cnnc(C)c1 c1(N2CCC(NC(CS(CC)=O)=O)C(F)C2)ncnc2sc(C(C)(C)C)cc12 C1(NC(C23CC(NS(=O)(=O)C(F)F)(C2)C3)=O)CCN(Cc2ccccc2)CC1 N1(C(C2C(c3ccn(C)n3)C2)=O)CC2CC(NC(=O)CCS(N)(=O)=O)C(C2)C1 C(=O)(CCCC(=O)NCCNS(=O)(=O)NC1CC(C(=O)O)C1)OCCCC(C)C N1(C(C(CC)=CCCC)=O)CCN(C(c2ccccc2SC)=O)C(CCO)C1 CCCCCCCCOCC(=O)NCC1(F)CC(NC(c2ccncn2)=O)C1 c1(C(=O)NC2C(C)CCN(C(COCC)=O)C2CC)nccc2ccccc12 CC(C)(CNC(=O)C=C1CCC1)NC(C1CC1c1cn[nH]c1)=O C12(Cc3nc(-c4c(OC(C)C)cccn4)nn3CC)CCCCC1C2(F)F C(=O)(CC(C)C(C)C)N(C(CNC(COc1ccc(SC)cc1)=O)C1CC1)C CON1CCC(CC(=O)NCC(C2CC2)NC(=O)CSCC2CCCO2)CC1 S(=O)(=O)(C1CCC(C(F)(F)F)CC1)NCCCC(C)(F)F c1(CCC)n[nH]c(=NC2CN(C(C3CCn4ccnc4C3)=O)CC3(CCC3)C2)s1 C1(CC(=O)NCCOC2CCCO2)CC2(CC2)CN1C(=O)COCC1CCOC1 C(C(C)(C)C(F)(F)F)NC(C1N(C(Cc2cc(C)no2)=O)CCC1)=O N1(C(CSCC)=O)CC(O)CC1C(N1CCC1n1cccn1)=O C(=O)(C(COC)CC(C)C)N1CC(C)CC(NC(C(C)NC(COC)=O)=O)C1 N1(C(C(C)=C(C)C)=O)CCN(C(C2CC(O)(c3ccccc3)C2)=O)C(C(F)F)C1 c1(N(C)C)c(COC(c2ccnn2-c2cccnn2)=O)cc(Cl)cc1Cl C1(NC(C(=O)NC2CC2)=O)CC2CCC(C1F)N2C(C1CNC(=O)N1)=O C1(CNC(CS(=O)(=O)NC)=O)CC2(CCC2)CN1C(c1cc(F)c(F)c(F)c1)=O C(C(CC(C)C)C(=O)N1CC2C(C1)C2(F)F)NC(c1nc(C)n(C)c1)=O c1(C(C)C)ncc(Cl)c(C(=O)NCCOCCCN(C(=O)CCC(C)(F)F)C)n1 c1(CC)cnc(C(=O)NCC(COC)OC)nc1.C1(=O)C(OC)CN1 c1(OC)ccnc(-c2ccc(=O)n(CC(N3CCC3c3ccccc3)=O)c2)c1 N1(C(C(C)C(F)F)=O)CCOC2CCN(C(c3cnn(CCO)c3)=O)CC12 c1(CN2CC(C)(CNC(c3c(CC)onc3)=O)C2)c[nH]c2c(C)cccc12 CC(CC(=O)N1CCCCC1CCNC(c1cncc2c[nH]nc12)=O)C(F)(F)F C1(C(N2CC(NC(=O)NC)C2)=O)(NC(C2CC(F)(F)C2)=O)CCSC1 CC(C)(C)C(C#N)C(=O)N1CCN(C(=O)COc2ccccc2)CC1C1CCC1 N(C1CCc2ccc(Cl)cc21)CC(C)(C)OC.c12ccccc1NC2=O c1(C(=O)NC2CC(NC(c3n[nH]cc3CC(F)(F)F)=O)C2)cn(CF)nn1.C(F)(F)F c1(CCCC)ccc(C(N2CC(NC(=O)C(C)C(F)F)C(O)C2)=O)cc1 C(c1nc2ccccc2s1)=CC(=O)N(C1CC(NC(C(C)(C)SC)=O)C1)C Cc1cc(CCCC(=O)NC2CC2CNC(C2CCC(C(N)=O)CC2)=O)c(C)s1 c1(CCC(=O)NC(C)CCCNC(c2nccs2)=O)ccc(C#N)cc1F c1(OCC)ccc(C(=O)NC2CC(F)CN(C(=O)C(C)SC)C2)c(F)c1F C1(C(N(C)CC2(CNC(CCC=C(C)C)=O)CC2)=O)CC(C)(C)OC1(C)C N1(C(C2N(CC#C)CCC2)=O)CCCC(N(C)C(C2C3C4CCC(C4)C23)=O)CC1 N1(C(C2(OC)CC2)=O)CC=CC1CNC(=O)C(O)CSCc1ccccc1 CCC(O)CC(=O)N1CCC(C)C1CNC(=O)CC1(NC(C)=O)CC1 C1(C)(NC(CC(C)(C)NC(=O)CCc2ccc(F)c(F)c2)=O)CCCCC1O c1(OC)cc(=NC(=O)C(C)(C)CN(C)C(c2cnsc2)=O)[nH]n1C S(=O)(=O)(C1CC2(C1)CC1(CCC1)C2)N1CCN(C)CC(CO)C1 Cc1cnn(CC(=O)NC(C2CC(NC(c3cscc3Cl)=O)C2)C)c1 c1(C(=O)NC2C(C)CCN(C(=O)CC3OCCO3)C2C)cn(C)c(=O)n(C)c1=O N1(C(c2c(C)oc(C(C)C)c2)=O)CCN(C(=O)C(C)(C)N2CCCC2)CC12CC2 C1(NC(C2CC(=O)N2)=O)CCN(C(=O)CCCC2CC2)CC1F C(=O)(C1CCCc2n[nH]cc21)N(CCCCNC(C1N(CCC)CCCC1)=O)C c1(OC)cc(C(N2CCN(CCCNC(c3ccon3)=O)CC2)=O)cc(Cl)c1O Cc1nc(C(N2CCOC(C(C)NC(=O)Cc3cnnn3C)C2)=O)c(C)s1 CC1(C)OCC2CC12NC(C1CCC(NC(c2ccccc2Cl)=O)C1)=O c1(N(C)CC)[nH]c(=NC(C)c2scnc2C)nc2c1ncn2C.C12CCN(C1)C2 C1(CC(=O)NCC2(CN(C(C(CNC(C)=O)(C)C)=O)C)CC2)CCOC(C)(C)C1 C1(NC(C(C=CC)O)=O)CCCCC1NC(=O)CC(=O)Nc1ccc(CF)cc1 CCC(O)C(C)C(=O)N1CCCCCC1C(=O)NC(c1nccc(O)n1)C C(c1nc(N(C)C)ncc1Br)C(Cn1nc(C)oc1=O)=O C(=O)(C1CCCn2c(CO)nnc21)NCCCNC(c1c(F)cccc1Br)=O C1(CC(=O)N(C2(c3ccccn3)CC2)C)CCCN(c2cccc(F)c2)C1=O C1(C(=O)NC(CCCNC(=O)CCN2CCC2)c2ccccc2)CC2C=CC1C2 c1(-c2cn(C(C3CCC(NC(C(CC)COC)=O)C3)CC)nn2)cc(C)cnc1F N1(C(CCS(C)=O)=O)CCC(n2cccn2)(C(=O)NCC2CCCCCC2)CC1 C1(NC(c2c(C)nc(CCC)s2)=O)CCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1 Cc1cc(Br)ccc1CNC(=NCC1CCN(C2CCCCC2)C1)NC1CCC1 c1(C(N(CCN(C)Cc2ccccc2Br)C)=O)ccc(-n2cccn2)nc1 c1(C(=O)NCC2C(NC(c3cnc(COC)s3)=O)CCCC2)cc(C#N)ccc1C C(=O)(CCCC(C)=O)NCC1N(C(CCCCC)=O)CC(C(F)(F)F)C1 C1(NC(=O)NC(c2ccc(N(C)C)cc2)C)Cc2nccnc2C1 N1(C(CC(OCC)OCC)=O)CCCC(CC)C1C(N1CC2(CCC2)C1)=O N1(C(C2CCCCC(=O)C2)=O)CC(NC(=O)Cc2ccc(Cl)nc2)C2CCCC12 C1(C(=O)NC2CN(C(C3(CC(C)C)CCCC3)=O)CC2F)CCCCC1(F)F C=CCCCC(C(=O)NCC1=NOCC1)NC(=O)CC1CC2CCC1O2 CC1CCc2[nH]c(C(=O)NC3(CNC(C4CNC(=O)C4)=O)CC3)cc2C1 CC1CN(C(c2cc(C(F)F)ncn2)=O)CC1NC(=O)CCc1cnn[nH]1 C1(CNC(c2c(CC)nn[nH]2)=O)CCC(F)(CNC(=O)C(C)n2cncn2)CC1 c1(CCC(=O)NC2CCN(C(c3cnnn3C3CC3)=O)CC2)ccc(O)cc1 Cn1cc(C(N2CCCC(c3ncc(C(F)(F)F)[nH]3)C2)=O)cc1C1CC1 c1(C(=O)NC(C(=O)OC)(C)C(F)(F)F)cnc2nc(Cl)ccc2c1 C1(OC)(CNC(=O)CCN2CCCCC2=O)CCN(C(=O)Cc2ccns2)CC1 c1(COC(C(c2ccc(C(F)(F)F)cc2)CC)=O)cc(Cl)ncc1F N1(C(C2CCN(C(C)=O)C2)=O)CC(NC(=O)CN2CC3CC3C2)C(S(C)(=O)=O)C1 C1(NC(c2c(C)nn[nH]2)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CCC2C1 N12CCN(CC1)CC2=O.C(C(C)(O)COCC#N)NC(C)=O C(CC(C)C)(C(=O)N1CCCC1CO)NC(c1cn(CC)nc1C)=O Cc1nc2cc(C(=O)NC(C)CCN(C(=O)C(CC(C)C)N(C)C)C)ccc2o1 Cc1ccc2c(c1)CC(C(=O)NCC1(CNC(C3CC34CCCCC4)=O)CC1)S2 C1(C(N(CC(=O)NCC2OCCC2C)CCC)=O)CCCCNC1=O N1(C(C(=Cc2ccncc2)C)=O)CCCC(CCNC(=O)C(F)C(C)(C)O)CC1 C1(CCC)CN(C(=O)C(COC)N(C)C)CCN1C(=O)Cc1cccnc1 C1(CNC(=O)CCC2(O)CCC2)CN(C(C2(CO)CCC2)=O)CCCO1 c1(-c2ccc(NC(C(CC#C)C)=O)cc2)cc(SC(C)C)ncc1C c1(CC(N2CC(N(C(=O)Cc3cn(C)nn3)C)C(O)C2)=O)cccc2[nH]ncc12 c1(C(=O)NCC2(NC(C(C)OC(C)(C)C)=O)CCOC2)cnn2c1OCCC2 c1(C(C)C)ccc(C(=O)N(C2CN(C(C3CNC(=O)N3)=O)C2)C)cc1 Cc1ccc2[nH]c(CN3CC4CN(C(c5ccnc(Br)c5F)=O)CC34)cc2c1 C(=O)(C1Cc2c(Cl)cccc21)N1CCN(C(c2cc(C#N)no2)=O)CC1CCO N1(CC)CC(C)N(NC(=O)OC(C)(C)C)C(C)C1C.c12cnccc1NC2=O N1(C(c2c(CNC(C3(CC)CNC(=O)C3)=O)c[nH]n2)=O)CCCC(O)(CO)CC1 Cn1ncnc1C(C)(C)NC(=O)CCOCCCNC(=O)C(O)Cn1cncn1 C1(N(C(C2C(=C)C2)=O)C)CCCCN(C(c2ccc(C(C)C)c(Cl)c2)=O)C1 C(=O)(C1CCc2ccccc21)NCc1nccc(C(=O)NCCn2cncn2)c1 N1(Cc2ncc(C)o2)CCC(NC(c2ccn(C)n2)=O)C(O)C1 C=C=CCCC(=O)NC(CCC)C(=O)NCC1(O)CCOC1C CCC(C(=O)N1CCC(OCC(=O)Nc2cncc(OC)n2)C1)C(F)(F)F O=C1CCC(C(=O)NCC2CC(C(N3CC(N4CCOCC4)C3)=O)CO2)O1 CCCC(C(=O)N1CC(OC)C(NC(=O)C(C)(C)n2cccn2)C1)S(N)(=O)=O CCCC(C)C(=O)N(CCCNC(c1cccc(=O)o1)=O)CC1CCCC1 CC(CN=c1[nH]cnc2cccc(F)c12)N(C)C(C1CC2(CCOCC2)CO1)=O C(=O)(C1=CCCN(C(c2c[nH]c(C(N)=O)c2)=O)C1)Nc1cn(CCC#C)nc1 C1(NC(CCCC)=O)CCCC(NC(c2cocc2Br)=O)CC1 n1(CCNc2ccc(C#N)cc2C(F)(F)F)cnc2ccccc2c1=O N1(C(C(C)Oc2ccc(F)cc2)=O)CC2CCN(C(=O)CCCN(C)C)C2C1 CC#CCCC(=O)N(CCCNC(c1cnc(CC)nc1C)=O)CC C(CCC(F)(F)F)N(C(Cc1cccc(F)c1)C(=O)Nc1cccc(Br)c1)C C12(C(=O)NCC3(c4ccc(OC)cc4)CCCCC3)CCCCC=C1OCC2 N#CC1CC2(CC(OC(=O)C=Cc3csc(C(F)(F)F)c3)C2)C1 C1(C(N(CC(C)NC(=O)CC2COCCOC2)C)=O)CCCCCN1C c1(NC(C(CC)NC(C)=O)=O)ccc(C(F)(F)F)cc1F.C12CCN(C1C1CC1)C2 c1(C(=O)NC(CC)CNC(c2cnncc2NC)=O)ccc2c(c1)CCC(O)C2 C(CS(=O)(=O)CCOCc1ccccc1)NC(C(CC)C)c1nnnn1C1CC1 CC1CC(NC(c2cc3occc3s2)=O)CCN1C(c1ccc(N)cc1Cl)=O N1(C(COC(C=C)=O)=O)CC(SC)CCC1=O.N1(CCO)CCN(C)CC1 C1(CNC(C2C(C)C2)=O)CCN(C(c2csc(C(F)(F)F)n2)=O)C12CC2 CC(CCN(C(=O)CCc1cnn[nH]1)C)NC(=O)CCSCC(N)=O CCC(C)C(CN(C)C)NC(=O)C(C1CC1)N(C(=O)C=CC(C)C)C CC1=C(CCNC(=O)C(C)(C)C2CCCN2C(=O)CC(C)C(C)C)COCC1 Cc1cc(C(=O)NCC(C)(C2CCC2)NC(=O)C2=CC(C)CC2)c2n[nH]cc2c1 N1(C(CC=C)=O)CCC2(CC(NC(=O)CCC(=O)NC3CC3)C2)C1 N1(C(C(CCC)C)=O)CC2CCCC(N(C(=O)CCc3ccc(F)cc3)C)C2C1 N1(CCCC2CCN(C(=O)C=CC(c3ccccc3)=O)C2)CC2CCC1CC2 C1(CNC(C(C)CN(C(=O)C=Cc2cccnc2)C)=O)CCC2(CC2)CO1 C1(OCC)CN(C(=O)C(c2ccc(F)cc2)(F)F)CC1CNC(=O)C=CC(C)C N(C1CCCn2ncnc21)C(CC(CNC(=O)C1=COCCO1)OC)=O c1(N2CCC(CCOC)(CO)C2)nccc(C)c1F C1(NC(CN2CCC(C)(O)C2)=O)CC2CC1CN(C(=O)CCc1ccncn1)C2 c1(C(=O)NC(CNC(c2c(OC)csc2)=O)C)cc(-n2ccnc2C)ccn1 N1(C(C=C(C)CN2CCCC2)=O)CCC2(C1)CN(C(c1csc(C)n1)=O)CCO2 CN1C(=O)CCCC1C(=O)NC1CCCCN(C(C2(O)CCSC2)=O)C1 N1(C(COCC#C)=O)CCOCC1C(=O)NCCN(CC(C)C)CCO N1(CCc2ncc(C)cn2)CCCC1C1CCCCN1C(=O)CC1CC=CCC1 C(=O)(CCCCOC)N(CC(=O)NCc1cc(COC)on1)CCC Cc1ccc(S(=O)(=O)C2(C(=O)N(C3CCN(C)C3)CC(C)C)CCCC2)cc1C c1(OC)ccc(C)cc1C(N1CCCC(NC(c2cc(C3CC3)nn2C)=O)C1)=O C(=O)(C(C)(O)C(F)(F)F)NCC(C(C)C)NC(C1(SC)CCC1)=O c1(C(N2CCC(O)(CN(C(Cc3c(C)noc3)=O)C)C2)=O)coc2c1COC2 Nc1ccc(C(N2CCC2CNC(C2CCCC(F)(F)C2)=O)=O)cc1N N1(C(CC(=C=C)C)=O)CCOC2(CCCN(C(c3ccc(Cl)cc3O)=O)C2)C1 C(=O)(C1CCCc2cc(O)ccc21)Nc1cn(-c2cc(COC)c(C)nc2)nn1 CC(Cc1ccnn1C)C(=O)NCC12CC(NC(=O)Cc3cncn3C)(C1)C2 N1(C(Cn2c(-c3cccc(OC)c3)ncc2)=O)C(C)CC(CC(=O)O)C1C N1(CC=CC(=O)N(C(C)C(=O)NCC#CC)CC=C)CCOCC1 C1(CNC(CSC)=O)CCCC(CNC(C2(c3n[nH]cc3C)CC2)=O)C1 CC1(C(=O)NCC(O)CCNC(c2cncc(N)c2)=O)CCCNS1(=O)=O c1(OC)ccc(F)c(C(=O)N(C)CCNC(C2CCN(C(C)C)CC2)=O)c1 CCCC(C#N)C(=O)NC1CCC(NC(=O)Cc2cccc(NC(N)=O)c2)CC1 N1(C(C(C)(C)CO)=O)C2CCC1CC(CNC(c1cccc(Cl)c1F)=O)C2 c1(C(C(=O)NC2CC(NC(COCCC(C)C)=O)C2)O)ccc(C2CC2)cc1 c1(N(C)C(C2COCC2NC(C2(Cl)CCC2)=O)=O)cccc(C#N)c1 c1(SC)nc(Br)c(C=O)s1.c1(CCC2CN(N3CCCC3)C2)cn(C)nn1 c1(-c2ccc(SC)cc2)cnc(NC(c2cn(C(C)(C)C)nn2)=O)c(O)c1 N1(C(C2(N(C)C)CCC2)=O)CCCC(CNC(=O)Cc2nn(C)cc2Br)C1 CC1(C)CCC(CC(=O)NCC2CC(NC(=O)C(C)(C)CCF)C2)CC1 Cn1c(C(=O)NCC(C2CCC2)NC(=O)CCNS(C)(=O)=O)cc2ccsc12 C1(N(C(C=COCC)=O)C)CCN(C(C2NC(=O)C3CC23)=O)CC1 Cc1ccc2oc(C(N3CC(SC4CC4)CC(NC(=O)CN(C)C)C3)=O)cc2n1 C1(C(=O)NCCC2(C)CC2)CCC2(CC2)N1C(c1cnc(C(C)C)o1)=O c1(N2CCC(NC(c3c(C(C)C)ocn3)=O)C2)nccc(S(C)(=O)=O)n1 c1(NC(c2nc(C(=O)NC3CCCO3)cs2)=O)cc(F)ccc1CC1CC1 C1(C(=O)NC2CCS(=O)(=O)CC2)CCN(C(c2cccc(O)n2)=O)CCO1 c1(CN(CCCN(C)C)C(C2(OC)CCSC2)=O)nc2cccc(C)c2s1 c1(CC)ccc(C(=O)N(CC(C)O)CCNC(C2CCSC2)=O)o1 C1(NC(C2(SC)CC2)=O)C(C)(C)CN(C(=O)C(C)NC(=O)C(C)(C)C)CC1(C)C C=CCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)CCc1csc(C)n1 CC1CCCC(CC(=O)NC(C)(C)CNC(c2cc(O)ncn2)=O)C1 C(=O)(CC(C)C(F)F)NC1C(C(=O)Nc2c(C)cccc2)CCC1 CC1CCC(C(=O)NCC=CCNC(=O)CC2CCCCC2)C1 CC(C)C(F)C(=O)N1CCC(C)(NC(=O)Cc2cccnc2)C1 C1(CNC(COCCC=C)=O)CC2CN(C(=O)C(N3C(=O)CCC3=O)CC)CC12 C(=O)(C(O)CC(F)(F)F)NCC1(F)CC(NC(c2ccc(C(C)(F)F)cn2)=O)C1 c1(NCc2cn(C)nc2C(F)F)cnc(O)c(F)c1 CCCS(=O)(=O)CC(=O)N1CC2(CNC(=O)CC(C)C)CC1(CC)C2 C12(NC(Cc3nc(C)sc3)=O)CCCC1N(C(c1cc([N+](=O)[O-])oc1C)=O)CC2 Cc1nc(C(=O)NCC2CN(C(=O)Cn3cnnn3)CC2C)c(C)o1 N1(C(C=CCN(C(C2C(C)CCCC2)=O)C)=O)CCC(C2CCCC2)C1 Cn1nc(C(N2CCC(O)(CNC(=O)CNC=O)CC2)=O)c2c1CCC(C)(C)C2 N1(C(c2nc(COC)oc2)=O)CCN(C(C2CC3C=CC2O3)=O)C(C)C1 N1(C(CC2CC(=C)C2)=O)CCCC1(C(N1CC(N2CCC2)C1)=O)CCCCO N1(C(C=CSC)=O)CCCC(C)(CNC(c2nnn(-c3ccccc3)c2C)=O)C1 CC1=C(C(=O)NCC2(CCN(C(=O)CCC3(C)CC3)CC)CC2)C(C)(C)CCC1 C1(C(=O)NC(C(C(C)C)NC(=O)CSc2nncn2C)C)CCCCC12CCC2 C1(C(=O)NCC(n2cc(CN3CC4CC4C3)nn2)C)CCC(=O)N1 C1(O)(CN(C(C2N(CC)CC2)=O)C)CN(C(=O)C(=O)NCC(F)(F)F)C1 C#CCC(C)(C)C(=O)NC1CC(C)N(C(c2c(-c3cccs3)noc2C)=O)C1 C(=O)(C(C)S(C)(=O)=O)N(C)CC1N(C(c2c[nH]c(=NC)s2)=O)CCOC1 Nc1cncnc1C(N1CCCCC1C(=O)NCCC1CC(O)C1)=O C#Cc1ccc(F)c(C(N2CCN(C(=O)CC3CCCCC3O)C(C)C2)=O)c1 c1(C(N2CCC(C)SCC2)=O)ccc2c(n1)CN(C(=O)CCCN=[N+]=[N-])CC2 N1(C(c2c(OC)ccs2)=O)CC(C)CN(C(C2CCCC23OCCO3)=O)C(C)C1 C12(CNC(C(c3ccccc3)OCC)=O)CC(NC(C3CC3F)=O)(C1)C2 c1(C(N2CCN(C(CCC(CC)CC)=O)CC2C)=O)ccc(S(=O)(=O)NC)nc1 CC1CC(CC(=O)NC2CCN(C(C3CCCOC3)=O)C2(C)C)CCC1C Cc1cccc2[nH]c(C(N3CC(NC(=O)CCCCN(C)C(C)C)C3)=O)cc12 N1(C(C)=O)CCC(O)(C2CCN(C(c3cc4ccc(Br)cc4o3)=O)CC2)C1 Cc1cc2nc(Cl)[nH]c(=NCC3(O)CCN(C(c4[nH]c(O)nc4C)=O)CC3)c2s1 c1(OCC)ccccc1C(=O)NC1CCC(C(=O)NC2CCN(C)C2=O)C1 C(=O)(CC(O)CCC(C)CC)NCCCNC(CCCc1ccc(C#C)cc1)=O c1(COC(C(n2c(C)cc(C(F)(F)F)n2)C)=O)ccc(Cl)cc1C(F)(F)F N1(C(C=CC(CC)C)=O)CCC2(CC1)CN(C(c1nc(Cl)oc1C)=O)C2C(C)C C1(NC(C(CN(C)C)O)=O)CC2CN(C(c3cnn(C)c3Br)=O)CC2C1 C1(C(C(=O)NCc2cccs2)N(CC(=O)OCC)C)CC2C=CC1CC2 N1(C(CCCC(C)C)=O)CCC(C)(C)CC1C(=O)NC(C)CC(C)C c1(NC(CCCNC(C2C(C)OC(C)C2C)=O)C)ccc([N+](=O)[O-])cc1F c1(C(=O)NC(C(C)(C)C)CNC(C2(C(C)(F)F)CC2)=O)cn2c(n1)CCC2 c1(C(N2C(CNC(c3n(CC)cnn3)=O)CCC2)=O)cc(C)ccn1 c1(C(N(CCCN(C)C(C23COCC2C3)=O)C)=O)ccc2sccc2c1 C(CC(=O)N(C)C)(C(=O)O)NC(c1ccc(Nc2ccc(OC)cc2)cc1)=O N1(C(c2ccn(C)c2)=O)CC2CC(NC(=O)CC3(C(F)(F)F)SCCS3)C(C2)C1 c1(CN(CC(CCCCN(C)S(N)(=O)=O)O)C)ccc2c(c1)CCN2C C1(C)(CC(=O)N(C)C)CCCN1C(C(=O)NCSc1ccccc1)c1nc[nH]n1 c1(C(N2CCN(C(CC(CCC)C)=O)C(C)CC2)=O)ccc2c(c1)OCCO2 C(c1cccc(Br)c1)=CC(=O)NCC(CC=C)NC(c1cnc(O)n1C)=O n1(CC)nc(CN2CCN(C(c3ccc(C(C)=O)o3)=O)C3CC23)c2ccccc12 N1(C(C2CC(C(C)(C)C)C2)=O)CC(CNC(=O)CN2CC3CC3C2)CC1(C)C c1(CC)oc(C(=O)NCC(c2ccccc2)NC(c2cnc(C3CC3)s2)=O)cc1C C1(NC(C2CCC(COC)O2)=O)CCN(C(=O)C#CC(C)C)CC1C C12(CNC(COCC)=O)CCCC1CN(C(C1(F)C3CCCCC13)=O)C2 c1(C(N(C)CCc2ccccc2Cl)=O)cc2cc(N)ccc2o1 N1(C(c2cc(CC)[nH]n2)=O)CC2CCC(NC(=O)C=CC(C)CC)(C2)C1 c1(CC(=O)NC(C2CN(C(C3(OCC)CCOC3)=O)C2)C)cn2c(C)csc2n1 c1(C(=O)NC2(C)CCN(C(Cc3cn(C(C)(C)C)nc3)=O)C2)[nH]cc2c1CCC2 C1(CNC(C(OCC)OC)=O)CCC2CN(C(=O)COCC3CC3)CC12 C(=O)(CC(C)CC(=O)NCC1CCN(C(c2ccc(Cl)c(F)c2)=O)C1)OC O=S(=O)(NCC1(OCCO)CCC1)N1CCCC(S(=O)(=O)N2CCOCC2)C1 C(=O)(CCCCC(F)F)NCC(CCOC)NC(C1CCCC1OC)=O C1(CC)CN(C(=O)CC(CC)CC)CCN1C(c1ccnn1CC#N)=O c1(C(C2CCOC2)OC)nc(-c2cc(C(F)F)on2)n(C(C2(C)CC2)C)n1 C(=O)(C(C)(C)Cc1cnn[nH]1)N(CC(C1C=NNC1=O)NCC(CC)CC)CC CC(CC(=O)NCC1CCCC1NC(=O)Cc1nc[nH]n1)c1cnn(C)c1 Cc1nc(C(=O)NCC23CC2CN(C(C2(C4CC4)CC2)C)C3)ccc1C(N)=O N1(C(C(CCC)F)=O)Cc2ccc(CNC(=O)Cn3ncc(Cl)c3C)cc2C1 c1(C(=O)NC2C(NC(C3N(C(C)=O)CCC3)=O)COC2)nccc(Cl)c1C C1(C(N2CC3C(CNC(CCC=CC)=O)C3C2)=O)CCc2nn(C)cc2C1 CC(C)CS(=O)(=O)CC(=O)N1CCCC(CN(C(=O)C2=CCCOC2)C)C1 C1(CCOCC)CCc2nc(NC(N3CCCCC3c3nc(C)cs3)=O)sc2C1 N1(C(C(CCC)CC)=O)CCC(C2CCN(C(c3ncc(N)cc3C)=O)C2)CC1 c1(C(N(C(n2cc(C(C)(O)CCO)nn2)(C)C)C)=O)occc1CN(C)C Cc1ccc(C(=O)NC(c2ccc(OC(F)(F)F)cc2)CO)c2c1CCC2 C12(CNC(=O)C3=CCCS3)CN(C(=O)Cc3cccc(F)c3)CC1CS(=O)(=O)C2 Cn1cc(NC(c2cn(CC3CCS(=O)(=O)C3)nn2)=O)c(C(F)(F)C(F)(F)F)n1 c1(OC)ccc(-c2nc(-c3nccn3C)n(C(C)C(C)(C)C)n2)cc1 C(=O)(CCCCCn1cnnn1)NC(C1CCCN1C(=O)CCCN(C)C)C C(C(=O)NC1CC(CCNC(c2cscc2SC)=O)C1)(C(C)C)OC c1(NC(C2N(Cc3ccc(N(C)C)cc3)CC2)=O)cc2c(cc1Br)OC(F)(F)O2 Cc1cc(C)c(C(=O)NCC(C)(C)NC(C2CCCC(O)C2)=O)cc1N CCC(CC)(CC)C(=O)N1CC(CN(C)C(C2(N(C(N)=O)CC)CCCCC2)=O)C1 CCCCCC(O)C(=O)N1CCN(C(=O)CC(F)F)CC1CC1CC1 C1(CCNC(=O)CNC(=O)CC(C)C)(SC)CCOCC1.C1(=O)C(C)(C2CC2)N1 N1(C(CC2C(C)=NOC2=O)=O)CC2(C1)C(NC(c1cc(C)ns1)=O)CCS2(=O)=O C=CC(C)(CCOC)C(=O)NCC(C)N(C(c1cscc1C(N)=O)=O)CC c1(C(=O)NC2C(C)CCN(c3c(F)cnc(C)n3)C2)ccc2nnn(O)c2c1 CCCCC(=O)NCCC1(O)CN(C(=O)CCSC2CCCC2)C1 C1(CNC(c2cc(C)sc2)=O)CC2(CO1)CN(C(=O)C(C)(C)c1ccncc1)C2 Cc1ccccc1C1CC1C(=O)NCC=CCNC(=O)CCc1cc[nH]n1 Cc1cc2c[nH]nc2c(C(=O)NCC(CO)NC(C2CCCCC2(F)F)=O)c1N c1(C(N2C(C)C(NC(=O)CC3CCC(=O)N3)CCC2)=O)cc2nc(Cl)ccc2s1 CON1CCC(CC(=O)NCCCN(C)C(C23CC4CC2C3C4O)=O)CC1 C1(CNC(C2=NOC(CNC(Cc3nc(CC)oc3)=O)C2)=O)CC2OC(=O)CC12 O=S(=O)(c1cc2ccccc2cc1Br)N1CCC2(CC1)CC(N1C3CNCC13)C2 c1(C(N2CC(N(C)C(c3cc(F)ccc3F)=O)C2)=O)ncsc1S(N)(=O)=O CC(F)(F)C(C)(C)C(=O)N1CC2(COC(CNC(=O)Cc3ccc(Cl)nc3)C2)C1 c1(C(=O)NC(CC)(CNC(c2nc(Cl)sc2C)=O)CC)ccc2ncncc2c1 C1(CCC)CCC(C(=O)Nc2nc(N3CCCC3)ns2)CC1 c1(C(=O)Nc2ccnc(N3C(c4ccc(F)cc4)CCC3)n2)ccc2occc2c1 c1(C(N2C(C(=O)Nc3c(C)nc(C)o3)CC(O)C2)=O)cc2ccc(Cl)nc2[nH]1 CC(C(=O)Nc1cccc(CNC(=O)CCn2cncn2)c1)C(C)(F)F N1(C(c2ccn(CCNC(CC3C(CC)C3)=O)c2)=O)C2C=CCC1CCC2 c1(C(N(C(C)C(=O)NCC23CCCCC2C3)C2CC2)=O)cccc(F)c1F N1(C(C=CC=CCC)=O)CCN(C(c2ccc(C(C)(F)F)cn2)=O)C(C)CC1C CC(C)(C)CCC(=O)N1CC(NC(=O)CCN2CCNC(=O)C2)C1 C1(CNC(C2(C#C)CC2)=O)C2CN(C(c3cn(-c4ccccc4)cn3)=O)CC12 c1(NS(=O)(=O)CC2CC23CCCCC3)ccc2ncc(Cl)c(Cl)c2c1 c1(OCCC(=O)N(CCNC(C2(C)CNC(=O)C2)=O)C2CC2)cc(Cl)cc(Cl)c1 C1(C(=O)NCC(C2CCC2)NC(Cc2cccc(OC)n2)=O)CC2(CCC2O)C1 C(=O)(CCCC(C)(C)C)NCCn1cc(CNC(C2C(OCC)C2)=O)nn1 c1(C(C(=O)NC(C)CC2CN(C(c3cnc[nH]3)=O)C2)OC)cnn(C)c1 N1(C(c2ccc(CNC(C=C(COC)C)=O)s2)=O)CC2OCC(CO)C2C1 c1(C(N2CCC(NC(C3CC(O)(CC#C)C3)=O)C2)=O)ccc(S(C)(=O)=O)[nH]1 c1(CN(c2ccccc2)C(Cc2ccc(C#N)nc2)=O)cc([N+](=O)[O-])c(F)cc1Cl c1(C(=O)NC23CC2CN(C(c2sccc2Br)=O)C3)n[nH]c2c1COC2 c1(C(=O)NC(CNC(c2n3cc(C)sc3nc2)=O)CO)cc2c(=O)[nH]ccn2n1 c1(CCC(=O)N(C(CNC(c2n(CC)ccn2)=O)C2CC2)C)ccc(Cl)cc1F c1(OC)ncc(C(=O)N(CCC(=O)NC(C2CCOC2)CO)C)cn1 C(=O)(C(CN=[N+]=[N-])NC(=O)CC(C)O)N1CCN(C(=O)OC)CC1 c1(NC2C(C)CCN(C(c3cccc(=S)n3O)=O)C2)ncc2c(n1)COC2 c1(CCC(N2CCC(CNC(CC(C)OC)=O)C2C)=O)ccccc1[N+](=O)[O-] N1(C(C2C(=C)C2)=O)CC(F)(F)CC1CNC(=O)C(C1CCOC1)OC C1(NC(c2c(C)nc(C)[nH]2)=O)CCC2(CCN(C(=O)C(=O)CCC(C)C)CC2)C1 CN1C(=O)CCC1C(N1CCSCC1CCNC(=O)Cc1ccco1)=O C(CC1CC1)(C(=O)NCC(C)CN(C(=O)C(=O)N(C)C)C)OC c1(C(N2CC(CCNC(c3cc(C)no3)=O)C2)=O)cccc2ncccc12 CCC(C)CCC(=O)N(C(CC(F)F)C(=O)NC1CCCN(O)C1=O)C N1(C(C(CC=CC)C)=O)CCOCC(NC(c2ccc(CC3CCC3)cc2)=O)C1 O=C(CCCc1ncco1)NC1CC(NC(C2CCC2)=O)C1 c1(CNC(C(C)C#N)=O)nn(C)c2c1CN(C(c1scc3c1CCCC3)=O)CC2 CN1CCC(C(=O)NC(Cn2ccnc2)CO)(NC(=O)C=C2CCCCC2)C1 c1(C(=O)NCC2CN(C(C3C(C=C)OCCC3)=O)C2)ccc2c(c1)CNC(=O)N2 N1(C(c2cc(CC)ncn2)=O)CC(C(N2CCOCC2C)=O)CC12CCC2 N1(C(C2(COC)CC2)=O)CC(NC(c2nc(OC)ccc2OC)=O)CC(O)C1 C1(OC)CN(C)C(C)(C(=O)N(C2CC(NC(=O)CSC)C2)C)C1 c1(C(=O)NCC2(O)CC(NC(=O)C(Cl)=CCl)C2)cc(O)nc(O)n1 CC1CCN(C(C2COC(=O)N2C)=O)C(C(=O)N(C2CCCC(O)C2)C)C1 CCC(CC(=O)NC(C1CC1C(N1CCCC(C(=O)NC)C1)=O)C)CC(C)C C12(C(=O)NCCOCCNC(C3(C)CCNC3=O)=O)CCC(C)(C1)OC2 C1(CC)CCCCC1C(=O)NCC1CCN1C(c1conc1C1(C)COC1)=O N1(C(c2c(C)cc[nH]2)=O)CC2CC1C2NC(c1cnns1)=O C1(C(N(CC(CC)O)C)=O)CN(C(c2nccn2C)=O)CC1(F)F c1(C(=O)NC2C(C(N(CC)Cc3cccnc3)=O)C2)c(Br)cc(Br)c(O)c1Br c1(CN(C)C(C2(C)CC2Br)=O)cccc(CNC(CCCn2c(C)ncc2)=O)c1 c1(CC)nnc2n1CCCC2C(=O)N(CCCNC(=O)C(C)S(N)(=O)=O)CC c1(C(=O)NC2C(C)CN(C(c3cnn(C)c(=O)c3)=O)C2)cccc2c1C(=O)CC2 c1(C2(C(OC(=O)CCNCc3ccccn3)CCCO)CCCC2)cccc(Cl)c1 Cc1cccc2cc(C(=O)NCC3CCCC(NC(C4CC(O)C4)=O)C3)cnc12 N1(C(CCCC#C)=O)CC2CC(NC(c3cc(Br)no3)=O)C(C2)C1 c1(C(=O)NC2CC(CC(=O)NCc3ccccc3)C2)ccc2[nH]nc(Cl)c2c1 C1(NC(CN(CCC)C)=O)CCC(N(C)C(c2cc(C3CC3)ccn2)=O)CC1 C12(CNC(C3CSCCS3)=O)CCC(CN(C(c3cc(F)c(O)c(F)c3)=O)C1)C2 c1(OCC(C)C)ccc(CC(C)NC(=O)N(CCS(C)(=O)=O)C)cc1 C(=O)(CCCCC(=O)NCCC1CN(C(=O)C2=CCCO2)C1)OC N1(C(C(C(C)C)C2CCC2)=O)CC(NC(c2cnn(CCO)c2)=O)CC(F)C1 c1(C)ocnc1C(N(CC(C)C)NC(COCC)=O)=O.NCC.C(CN(C)C)O C1(c2cn(CC(=O)NCC3(C)CC=CC3)nn2)CCC(F)(F)CC1 N1(C(CCc2c(C)cccc2)=O)CCCN(C(=O)CCc2ccsc2)CC1 c1(C(=O)NCC2C(NC(C(C)(C)C3CC3)=O)C2)c(F)ccc(S(C)(=O)=O)c1F c1(C(=O)NC2CN(C(=O)CO)C3CC23)cc2nccn2c(O)n1 C1(C(N(C2CCN(C(=O)CCC3CCN(C)C3)CC2)CC)=O)CCC(C)(C)OC1 N1(C(CCC#CC)=O)CCC2(C1)CN(C(=O)C(O)C(C)(C)C)CC(C)O2 N1(C(C=C(C)Cl)=O)CCOC(C)(CNC(=O)Cn2cc(CN(C)C)nn2)C1 C1(CN(C(C2C(CN(C)C)C2)=O)C)CCC(CNC(=O)C=CC(F)(F)F)CC1 c1(OC(=O)C(C)Oc2cccc(Cl)c2)ccc(-c2ccc(COC)s2)cc1C C12(NC(C=C(CCC)C)=O)CCCC1CN(C(c1ccn3cncc3c1)=O)C2 CC(CSC(F)(F)F)C(=O)NCC(F)CNC(=O)C(c1ccccc1)O C1(CC(N2CC(CCC)OCC2)=O)C2CCCC2N1C(C1CC12CCOCC2)=O CCC(F)(F)CC(=O)NC12CC1CN(C(=O)CN(C1CCCC1)C)C2 C=C(C)CC(C(=O)N(CC(C)NC(c1cc(O)nc(O)c1)=O)C)NC(C)=O C1(NC(c2cc(COC)on2)=O)CCCN(C(=O)CCCC2CC2)C1C N1(C(c2c(OC)cc(C)cn2)=O)C2CCC1CN(C(c1coc(C(C)C)n1)=O)C2 C(c1ccncc1)=CC(=O)N(CC(CN(C(CN(CCCCCC)C)=O)CC)C)C N1(C(c2c(C)c[nH]c2)=O)CC2CC(NC(C3CNC(=O)N3)=O)C1C2 N1(Cc2cc(OC)cc(Br)c2)CCC2CN(C(=O)CCn3nc(C)cc3C)CC12 c1(C(N2C3CC(NC(C(COC)O)=O)C2CC3)=O)ccc([N+](=O)[O-])cn1 C1(NC(c2n[nH]c(C)c2[N+](=O)[O-])=O)CCOC12CCN(C(c1nncs1)=O)CC2 C(=O)(C(C)C(=O)N(c1ccc(CO)cc1)Cc1nc(C)cs1)OC C1(C(=O)NCCNS(CCC)(=O)=O)CC1C1CN(C(=O)OC(C)(C)C)C1 N1(C(Cn2c(C)nnn2)=O)CC2CC2(NC(C2COCC2(C)C)=O)C1 N1(CCCNC(C2CC(Br)C2)=O)CCCC(O)C1c1ccccc1 c1(C(N2CCC(NC(C(c3c(OC)cccc3)C)=O)CC2)=O)cccc(O)c1F Cc1c(C(=O)NC(C)CC(C)NC(c2cnn(C)c2Br)=O)ccn1C C12(C(N(C(C)C3CC3)C)=O)CCC(CC1)N(C(C1CNC(=O)C1)=O)C2 c1(N(CCN(C(C2CCN(C(CC=C)=O)CC2)=O)C)C)ccn2ccnc2n1 c1(C(=O)N(CC(N2CCCC2CNC(C2C3COCC23)=O)=O)CC)cccc(F)c1 C1(NC(c2cc(SC)oc2)=O)CCOCC1NC(=O)CCOC(C)C c1(C(=O)NC23CC(CNC(C45C(C)OC(C)(C4)C5)=O)(C2)C3)cc2cccnc2[nH]1 Cc1cc(N2CCC(CNC(=O)C=CC(N)=O)CC2)n2nc(C(F)(F)F)nc2n1 c1(C(=O)NCC2CC(NC(c3cnn(CC)n3)=O)C2)cccc2c1ccn2C c1(OC)cc(C(N2CC(CNC(C3CC4CCCC4C3)=O)(OC)C2)=O)ccc1O C#CC1(C(=O)N2CC=CCO2)CCN(C(c2cnn(CCC)c2)=O)CC1 Cc1ncc(NC(C2C=CC(NC(c3cc(Br)cnc3C)=O)C2)=O)cc1F c1(CCNC(COCC)=O)occc1C(=O)N(C(C)C(C)C)CC C1(NC(C=CC=CC)=O)CN(C(C2CC23CCOCC3)=O)CCC12CCOCC2 CC(C)C(F)(CNC(c1cc[nH]c1)=O)C(=O)NCC1CC2(CCC2O)C1 c1(C(N(CCCNC(c2cnc(Cl)cc2N)=O)C)=O)coc2c(Cl)cccc12 C(=O)(C(C)(C(C)C)NC(c1ccc(C(=O)O)c(C)c1)=O)NC C1(NC(C2(C)CCCN(C(C3CC4(CCO3)CC4)=O)C2)=O)CC2(C1)CC21CCC1 c1(OC)ccc(O)c(NC(=O)NC(Cc2ccccn2)CO)c1 c1(NC2C(C)(C)C(NC(c3coc(CC4CC4)n3)=O)C2)ncc(Br)cc1C#N N1(C(CSC(=N)N)=O)CCC2CN(C(c3cccc(C4CC4)c3)=O)CC2CC1 c1(C(=O)NC(C2(O)CN(C(=O)Cn3ncnn3)C2)C)ccc(Br)c(F)c1 C(CCCC(=O)N1CCN(C(=O)CNC(=O)CC2CCCC2(F)F)CC1)SC c1(C(N2CC(OC)C(NC(C)=O)C2)=O)ccc(Cl)cc1NC(=O)C=CCO O(N1CCC(CC(N2CCC(C)C2CNC(=O)CC(C)CC)=O)CC1)CC C(=O)(C1=C(Cl)CCOC1)N1CC(C(C)C)N(C(=O)CC2CCC23CCC3)CC1 C=C(Cl)CCC(=O)N1CCOCC1CC(=O)NCCCOC(=N)O c1(OCC)ccccc1C(=O)NC1CC1NC(=O)C(c1cccc(Cl)c1)C C12(C(=O)NC3CC(NC(Cn4nnc(C)n4)=O)C3)CCC(CO)(CC1)C2 C=CCC(C)(C)C(=O)N1CC(O)(CNC(C2(C(F)F)CCCC2)=O)C1 C12(NC(C(CSC)C)=O)CC(CNC(c3coc(Cl)c3)=O)(C1)OC2(C)C Nc1ccc(-c2nc(C3CC3(F)F)n(CC3NC(=O)NC3=O)n2)cc1 C1(C(=O)NCC(O)C2CC2)CCN(C(c2cc(C3CC3)ccn2)=O)CC1 c1(C(N2C(CCNC(c3c(C)nc[nH]3)=O)CSCC2)=O)cn2ccc(F)cc2n1 N1(C(=O)COc2ccnc(Cl)n2)CCN(C(c2ccsn2)=O)C(CO)C1 c1(CSC)ccc(Cl)c(C(=O)NC2CC2CNc2nc(C(C)C)cc(SC)n2)c1 CC1C(NC(C2CCCC(=O)N2)=O)CCCN1C(=O)COC1(C)CCCCC1 Cc1ccc(C)c(OCC(=O)NCC(C)N(C)C(C2CC(=O)CC23CC3)=O)c1 C(=O)(CC(C)C(C)(C)C)NCC(C)(Cn1cccn1)NC(CCCC=C)=O c1(OC)ccc(Br)c(C(=O)NCC(C)CNC(=O)C(C(C)O)NC(N)=O)c1 c1(NC(c2cc(OCC)ncc2-c2ccc(C)nc2F)=O)c(F)cc(F)cc1Br c1(C(=O)NC2C(CNC(C3CC(OC)C3)=O)CC2)c(C2CC2)cccc1F C1(C(N(CC(=O)OC)C2CC2)=O)CC(F)CN1C(=O)Cc1nccc(C)n1 C(C1CCc2nccn21)NC(C1(CC)CCN(C(=O)C=C2CCC(C)CC2)C1)=O N1(C(CCC(C)(C)NC(c2c(C)ccnc2C)=O)=O)CC(C)(C)C2COCC12 c1(NC(C2N(C(CC#C)=O)C3C(C2)C3)=O)cc(Cl)c(Cl)cc1Cl C1(O)CC2CC(C1)N(CC)C2.C=C1CC(C(=O)OC)N(C(=O)OC(C)(C)C)C1 C(CC(F)Cn1cc(C(C)O)nn1)NC(CNC(CCC)=O)=O CCC(CCCC(=O)N1CC(N(C)C(=O)OC)C1)NC(c1cnsn1)=O C1(NC(CC(COC)C)=O)CN(C(=O)C(C)(F)F)CC2CCCC12 C1(NC(C(C(C)O)C)=O)(CO)CCCN(C(=O)C(C)Cc2ccco2)C1 Cc1cc(F)ccc1C(=O)NCCCN(C(=O)C(F)C(C)C)C(C)C c1(CC(C(=O)NCC(C(=O)OC)C)C)ccc(Br)cc1.C12CC(C1)NC2=O C(=O)(CC(C(F)F)NC(c1ncn(C)n1)=O)NCc1nccc(OC)c1 C#Cc1ccc(C(N2CCCC2C2(NC(=O)CSC3CC3)CC2)=O)c(F)c1 c1(C(N2CCCC(NC(C=C(CC)CC)=O)CC2)=O)cc(F)c([N+](=O)[O-])cc1F C(=O)(CC(C)(C)C(F)F)N(CC(C(=O)NC1(CC=C)CCOC1)C)C c1(C(C2CCN(C(CSCc3nc(C)sc3)=O)C2)O)ccccc1F n1(CC(=O)N(C(C)C)CCNC(C2CCC2(C)C)=O)ncc(O)nc1=O c1(C(=O)NCc2ccc(F)nc2)cc2cccc(-c3cc(C4CCC4)n[nH]3)c2[nH]1 N1(C(Cn2nnc(C)n2)=O)CCC2CCN(C(c3nccc(Cl)c3F)=O)C2C1 C=CCC(C(=O)NC(C)COCC)NC(C1C(C)(C)C1(F)F)=O C1(NC(C(C)CCO)=O)CC2CN(C(=O)Cc3cc[nH]n3)CC12 N1(C(COC(CC)(C)C)=O)CC(O)CC1C(=O)NC(C)Cc1nc[nH]n1 c1(CC(N2C(CCNC(C3C(CC)CCO3)=O)CCCC2)=O)c(O)ncnc1O C1(NC(=O)CC2CCCCC2)CC(NC(c2csc(CO)n2)=O)C12CCOCC2 N1(C(C(F)OC)=O)CC2CC(C1)C2NC(c1cc(Cl)cc(Br)c1)=O n1(CC)nc(C)cc1C(=O)NC1C2CN(C(=O)C(C)N(CC(F)(F)F)C)CC12 n1(CC(=O)N(C)CC2CN(C(C3C(CC(C)C)C3)=O)C2)cc(CN(C)C)cn1 C1(c2cccs2)(C(CCC(=C)CNC(=O)C(C)(C)OC(C)C)=O)CCOCC1 c1(NC(C2CCC(C(=O)OCC)C2)=O)ccc2c(c1)nnn2C CC(C(=O)N1CCN(C(=O)CNC(c2cn3ccnc3s2)=O)CC1)S(C)(=O)=O CC1CC(C(=O)NCC=CCNC(c2cc(-c3ccco3)on2)=O)CCO1 C1(CC(=O)NC)CN(C(=O)C(C)Cc2ccccc2C)CCN1C(=O)CS(C)(=O)=O C1(C(=O)NCCN(C(CC(C)C2CC2)=O)C2CC2)CC(Cc2ccccc2)=NO1 Cc1nn(C)c(Cl)c1C(=O)NC1CCN(C(=O)C(C)C#N)C(C)C1 Cc1nc2cc(C(=O)N(C3C4CN(C(=O)C(C)c5ccco5)CC34)C)cnc2s1 N1(C(c2c(Cl)cc(C)nc2)=O)CCC2CN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2C1 N#CC1=C(C(=O)NC2C3CN(C(c4c(F)ccc(Cl)c4N)=O)CC23)CCC1 c1(C(=O)NCC2COCCN(C(c3ccc(C)s3)=O)C2)c(C)nc2ccccn12 c1(C(C)=O)ccc(NC(C2CCN(C(C3CC3(C)C)=O)C2)=O)c(F)c1 c1(C(N2CC3C(NC(c4cc[nH]n4)=O)CC(C3)C2)=O)cnn2ccc(Cl)c(F)c12 N1(C(C2CN(C(CCN(CC)CC)=O)CC2(C)C)=O)CC2CN(C)CC2(C)C1 N1(C(CC(CC)NC(CC=CC)=O)=O)CCc2c(cnn2C)C1 N1(C(Cc2ccc(C)s2)=O)CCOCc2cc(CO)ccc21 N1(C(C=CC=CCC)=O)CCC(C)(C)C(CNC(C2(NC(C)=O)CCC2)=O)C1 c1(C(=O)NC2CCN(C(C(C)(C)OC)=O)CC2C)c[nH]c2cnccc12 c1(OC)ccc(CN(C)CC2CN(C(C3CCNCC3OC)=O)C2)cc1F c1(C(N)=O)cc(NC(C2CC(O)CN2Cc2ncc[nH]2)=O)ccc1[N+](=O)[O-] N1(C(C(C)N2CCC2)=O)CC2CC(C1)N(C(C13CCCC1C3(F)F)=O)C2 N1(C(CC2CCCCC(=O)N2)=O)CCC2(CC1)CCN(C(C13CC(CO1)C3)=O)C2 Cc1cc(C(F)(F)F)nc(N2CC(N(C)C(c3cccc(O)c3C)=O)C2)n1 c1(CC)ccc(C(=O)NCC2(F)CCN(C(=O)CCN3CCCC3)C2)cc1Cl Cc1ccncc1CNC1CCC(C(=O)Nc2cccc(CF)c2)C1 C1(C(=O)Nc2ocnc2C(N2CC(=C(F)COC(C)(C)C)C2)=O)COC(C)(C)CO1 N1(C(c2cncc(-c3cccc(C(=O)OC)c3)c2)=O)CCC(O)C(F)(F)C1 CC1(C)C=C(C(=O)NC(CNC(c2ccn(C3CCCC3)n2)=O)CO)C1 C(=O)(C(=O)CC(C)C)N1C(CC)C(NC(=O)Cn2ccnc2C(C)C)CC1 C1(C(N2CC(C(C)C)C(C(=O)NCC(Cl)Cl)C2)=O)CN(C)CC(C)O1 N(C(=NCCC(C)C)N1CCC(CC(=O)NCC)C1)CC(=O)NCC=C CCCCC(C(=O)N1CCCN(C(C2CCC(C3CC3)CC2)=O)CC1C)C(C)C c1(OCC(N2CC(N(C(C(CC=CC)CC)=O)C)C2)=O)c(F)c(F)cc(F)c1F C=CCCCC(=O)NC1CC(C(=O)NC2CCN(Cc3ccc(O)cc3)CC2)C1 c1(C(=O)NC2(CN(C)C(C3(O)CCSC3)=O)CC2)ccccc1SC(F)(F)F C1(NC(c2cc(C)n(C(C)C)n2)=O)CN(C(=O)C2=NOCC2)CC1N=[N+]=[N-] C1(N(C(=O)CSCC2CCCO2)C)CCCCN(C(=O)C=C(C2CC2)C2CC2)C1 O=C1CSc2nnc(N3CCN(CC(N4CCCCC4)=O)CC3)cc2N1 O=C(N=c1cc(Cl)cn[nH]1)c1nc(-c2cnc(Cl)c(Br)c2)cs1 C(CC(F)F)(C(=O)N1CCOC(C2CC2)C1)NC(c1nc[nH]n1)=O C(=O)(CC(F)(F)C(F)F)NC1C(C)CN(C(=O)CCc2ccncn2)C1 CCC(C)C(C(=O)N1CC(C)C(C)(CNC(c2n[nH]c(C)n2)=O)C1)OC C=CCCCCC(C(=O)NC(C)(C)C)N(C)N(c1nccs1)C(C)=O CCCCCC(=O)NC1CC(F)(CNC(=O)CNC(=O)COc2ccccc2)C1 c1(C(=O)NC2CC(NC(C3C(C)C3(F)F)=O)C(O)C2)ccc(N)c(O)c1 C=C1CCN(C(C2CCNC(=O)C2)=O)C(C(=O)NCc2cncc(OC)n2)C1 C(CC(CC)C(=O)N(c1ccc(OC(C)C)cc1)C1CCCCC1)=CC N1(C(=O)Nc2cn(-c3cnn(C)c(=O)c3Br)nn2)CC2(CCNC2=O)C1 C1(CNC(c2c(CC)n[nH]c2)=O)CN(C(C2(C)CC2(C)C)=O)CC1(C)C Cc1ccc(C)c(C(=O)Nc2nc(CC(=O)NCCc3ccccc3C)cs2)c1 c1(OC)cc(CN2CCCC(C(=O)NC3(C)CCCCC3)C2)cc2c1OCO2 c1(OC)ccc(CC(=O)NCC(O)CN(C)C(C2CC2SC)=O)cc1F c1(OC)cccc(C(=O)NC(CNC(c2coc(O)n2)=O)C(C)(C)C)c1C C1(C(C)O)COCCN1C(=O)CC1CCN(C(c2nc(C(C)C)oc2C)=O)C1 C(=O)(CCCCCC(C)C)N1C(C(=O)NCCOCCCC#C)C(C)(C)CCC1 c1(C(=O)NCC(CNC(CC2C(C)C(=O)CC2)=O)O)cc(O)nc2c1CCCC2 N1(C(C(=O)OCC)=O)CCCC(CCOCCN(C(=O)CN(C)CCO)C)C1 C(=O)(C1=CCCOCC1)NC(CSC)(C)C(=O)NCc1cnc(C)c(C)c1 CC1(C)CC(C(=O)N2CCN(C(=O)CCC(N)=O)CC2CF)c2ccccc2O1 N1(C(c2c(C)onc2)=O)CC2CCC1C(C(=O)Nc1cccc(O)n1)C2 c1(C(=O)NC2(CNC(=O)C3CC3)CC2)cc2cc(Br)ccc2oc1=O C12(CNC(=O)CSc3ncc[nH]3)CC1CN(C(C1CN(C3CCOCC3)C1)=O)C2 c1(CC(N2CCN(C(C3CCCC34CCC4)=O)CC2)=O)ccc2c(c1)OCO2 c1(CNC(CNC(C)=O)=O)cccc(CN(C)C(c2cc(C)c(C)[nH]2)=O)c1 c1(OC)ccc2c(C(N3CC(C)(NC(c4cc(C)cnc4C)=O)C3)=O)csc2c1 CCCCC(O)Cc1nc(C(C)C)nn1-c1ccccc1CC c1(C(=O)NC2CN(C(=O)C=Cc3cccnc3)CC2F)ccnc2ncccc12 c1(C(N2CC(CC=C)(NC(=O)CO)C2)=O)cccc(C(C)=O)c1 C1(C)(CC)CC(C(N2CCOCC(CNC(c3cn(C)cn3)=O)C2)=O)CCO1 CN1C(=O)CCC1(C)CNC(=O)C(C1(O)CCC1)NC(=O)CC1CCC(O)C1 C1(NC(C2(CC#C)CCOC2)=O)CN(C(=O)CCn2ccnn2)CC(F)(F)C1 N1(C(C(=O)NC(CC)C(F)(F)F)=O)CCCCCC1c1ccccc1 C(=O)(CC(C)O)NCCN(C(=O)C(C)(C)c1ccnnc1)CC CC(C(=O)N1CC(O)CC1C(=O)N(c1ccccc1)C)C(F)F CCC(F)(F)CC(=O)N1CC(CNC(=O)CCc2nc(C)no2)C(F)(CO)C1 Cc1ccc(C(=O)N(C2(C(=O)NCC3CCCN(C)C3)CCC2)C2CC2)c(F)c1 C(=O)(C(CNC(c1cc(C)co1)=O)C(C)(C)C)NCC(C)(CO)OC C(=O)(C(O)CC(C)C)N1CC(OC)(CNC(=O)Cn2nc(C)oc2=O)C1 C(CC(O)CCO)NC(CCN(C(CCc1onc(C)n1)=O)C(C)C)=O N1(C(c2ccc(OC)nc2)=O)CC(C)(C)CC1C(=O)NC(C)C(C)(C)CO C1(C(N2CC(OC)C(NC(=O)CCc3ccc(C)cc3)C2)=O)CCC(C)(C)CC1 n1(CCC)ccc2cc(NC(C3CC(OC)CCO3)=O)ccc12 c1(NC(C2CCCN2CC2CC(F)C2)=O)ccc(Cn2ccnc2)cc1 Cc1ccc(-c2cn(C(C)CNC(=O)Cc3csc(NS(C)(=O)=O)n3)nn2)cn1 C1(NC(C2(CC=C)CCCCC2)=O)CCN(C(=O)CC(C)(C)C#N)CC1F N#CC1CN(Cc2ccc(O)c(Br)c2)CC1NC(c1csc(Cl)n1)=O CCCCC(C)(F)C(=O)NCC(O)CNC(C1(C)C=CCCC1)=O N1(C(CCC=CC)=O)CC2(COC(CNC(=O)C=Cc3ccncc3C)C2)C1 CC1CCCc2c(C(N3CCCN(C(C4COC(=O)O4)=O)CC3)=O)cnn21 C1(C(C)C)CN(C(=O)CC2CCC2)CCC1NC(c1ccn(C2CCC2)n1)=O C#Cc1cc(F)c(C(=O)NC2CN(C(=O)CC=C)CC2C)c(F)c1 N1(C(C2=CCN(C(C(COC)(C)O)=O)C2)=O)CCOC2(CCCC2)C1 C(=O)C(C)CC(C)C.C=C(C)COC(C)C C12(NC(=O)Cc3csc(Cl)c3)CCCN(C(c3nocc3Br)=O)CC1C2 CCCCC(C(=O)NCC(C)(C)CNC(c1cccc(F)c1Cl)=O)NC(N)=O C1(NC(C(COc2ccccc2)OC)=O)CCCN(C(c2ccc(O)nn2)=O)C1 CC1CCCC(C)N1c1ccc(SCc2cn(C)nn2)c(C(=O)O)c1 CCCC(C(=O)N1CCC(COC(N)=O)CC1)N(c1ccc(Cl)cc1)C c1(OC)cc(OC)c(N)c(C(=O)NC(C)CCNC(=O)C(C)C(C)(F)F)c1 C1(C)(C(=O)NC2CCN(C(C(c3ccc(C)cc3)(F)F)=O)C2)CCC12CCC2 C(=O)(C(C)C(F)(F)F)NCC1CC(COC)CN1C(c1cscc1C)=O C(=O)(CC(C)(C)C(=O)NCC1CN(C(C2CCCN2C)=O)C2(CCC2)C1)OCC c1(CNC(CN(C(C=CC(CC)C)=O)CC2CC2)=O)cccc(C)c1F CC(C)CCCC(=O)NCC1CC(C(=O)NC2CCCN(CCO)C2)=NO1 c1(C(N(CC(CN(C(c2cc(C)nc(O)c2)=O)C)O)C)=O)cc(F)cc(C)c1N N1(Cc2nc(N(C)C)oc2)CCCCCC1C(=O)O Cc1cc(Cl)cc2[nH]c(C(=O)N(C)CC3CCCN(C(=O)C(C)(Cl)Cl)C3)cc12 C1(C(N2CC=CC(NC(=O)CCC3CCCCC3)C2)=O)CC2(C1)CS(=O)(=O)C2 CC1c2ccccc2OC1CNC(c1cc2c(Cl)cncc2s1)=O N#Cc1cc(S(=O)(=O)NC23CC(C(=O)Nc4cc(Br)cc(I)c4)(C2)C3)ccc1Br CC1CCN(C(c2cnn(C)c2)=O)CC1NC(C1(C)CCC12CCC2)=O N1(C(C(C(C)C)O)=O)CC2C3CCC(C2C1)N(C(=O)CCc1ccc(Cl)s1)C3 C(C(C)CC(F)(F)F)NC(C1C(CC)N(C(c2ccncc2CC)=O)CC1)=O CCC(C)CC(=O)NCCC1CCN(C(=O)CCOCC(F)F)CC1 C#Cc1ccc(CN2CC3CC2CN3C(=O)C(c2ccccc2Cl)C)nc1 c1(CC)cc(C(=O)NC(C)Cn2cc(CNC(=O)CC(C)N(C)C)nn2)sc1C c1(CC(=O)NCC)csc(C)n1.C1CC(=O)N1CC(C(=O)OC)C1CC1 N#Cc1cccc(CN(C(c2ccc(Cl)cc2)C(=O)O)C2CC2)c1 C1(C(=O)NC(c2cnccn2)C)CN(C(c2cc(O)n(C)n2)=O)CC12CC2 c1(OC)ccc(CNC(=O)CCN(C(c2c(CO)cnn2C)=O)C2CC2)nc1 C1(N(C)CC)CCN(C(=O)C(C)(C)C2CCCN2C(C2OCCC2CC)=O)C1 c1(C(=O)NCC(=C2CN(C(c3[nH]cc(C)c3)=O)C2)F)ccc(F)c(C)c1 c1(C(N(C2CCN(C(c3cc(Cl)no3)=O)C2)CC)=O)csc(F)c1 C(=O)(CCCCCNC(C1(C)CCCN1C)=O)NCC(CC(=O)OC)O CCC(O)CC(=O)Nc1c[nH]nc1C(=O)N(CC)Cc1c(C)noc1C CCC(O)C(C)C(=O)N1CCC(CCNC(=O)Cc2cc(Cl)n(C)n2)C1 Cc1csc(S(=O)(=O)N2CC3CC3(C(=O)NC(c3cccnc3)C)C2)c1 c1(CC)cc(Br)c(C(c2nnnn2C)NC2CC(O)(c3ccccc3)C2)s1 c1(C(N2C(C)CC(NC(c3c(CC)c[nH]n3)=O)C2)=O)cccc2c1CCC(=O)N2 N1(C(C2(NC(C(c3cnn(C)c3)C)=O)CC2C)=O)CCC2CCCC2CC1 c1(CNC2CCC(CNC(c3c(F)cncc3F)=O)CC2)ccc2cc[nH]c2n1 N1(C(c2c(F)ncc(OC)c2)=O)CCCCCC(Nc2nc(C)nc(C)c2F)C1 c1(NCCc2c(OC)cccc2)[nH]c(=NC2CCCC2C#N)nc2sccc12 N1(C(C(C)(C2CCC2)NC(=O)C=CC2CCC2)=O)CC(CO)C2(CC2)C1 N1(C(c2cc(Br)co2)=O)CCC2CN(C(=O)C(O)CC(F)(F)F)CCC12 C#Cc1cccc(C(=O)NC2CC(C)N(CCOC)C2)c1 Cc1nc2cc(C(N3CC(C)(CNC(c4cc5n(n4)CCCC5)=O)C3)=O)ccc2s1 Cn1nnc2c1C(C(=O)NCCN(C(C1CC13CC(F)(F)C3)=O)C1CC1)CCC2 C(CCCC(=O)N1CCC(C(C)(C)CNC(c2oncc2C)=O)CC1)OCC c1(CCC(=O)NCCN(C)C(c2ccc(SCc3ccco3)o2)=O)c[nH]c(=N)[nH]1 C1(C(=O)NCCCCC=C)CCN(C(=O)C(=O)N(C)C)CCO1 c1(C(C)C)cc(NC(=O)NC(c2cccc(C(F)F)c2)C(F)(F)F)ccc1F N1(C(c2ccc(C)s2)=O)CCCC1C1CCCN1C(=O)COCCOCCO N1(C(C(CC)N2CCCC2=O)=O)CCCC(CN(C(=O)C(C(C)C)SC)C)C1 CC(C(F)(F)C(F)(F)F)=CC(N1CC(C)(C)CCC1CNC(C1CCSC1)=O)=O C(=O)(CC1=CCCC1)N1CC(CNC(CC(CC)C)=O)C1 C1(C(=O)NCC2C3CN(C(=O)C4=NOCC4)CC23)CCC2(CC1)CC2 c1(C(C)(CO)NC(=O)NC2CC3CCC2C3)cccc(F)c1 C1(CNC(COCC#C)=O)CN(C(c2cc[nH]n2)=O)CCC12CCOCC2 N1(C(C(C=C=C)C)=O)CC2(C1)CN(C(c1ccnn1C)=O)Cc1ccccc1O2 N1(C(C(CC)(C)C)=O)CCN(C)C(CNC(=O)C(c2ncccc2C)(F)F)C1 C1(N(C(Cn2ncn(C)c2=O)=O)CCCN(C)C)CC2(CCNCC2)C1 C12(NC(c3ccc(CC)nc3)=O)CC(C)(C1)OC21CN(C(=O)C(C)(C)CC#N)C1 C(=O)(C(C)(O)C(C)C)NCC1(O)CN(C(c2ccc(SCC)nc2)=O)C1 Cc1nc2ncccc2cc1CC(=O)N(C1CN(C(=O)C(C)(Cl)Cl)C1)C c1(-n2cc(CCOCC(=O)Nc3csc(Br)c3)nn2)ccc(F)c(Cl)c1 CC1CCCCC1C(NOC(c1cc(COCc2cccc(Cl)n2)[nH]n1)=O)=O Cc1nc(S)nc(C)c1CCC(=O)NC(C)(CNC(C1CCC(=O)O1)=O)C(C)C CC1CCN(C(=O)C(C)(C)C(N)=O)CC1NC(c1ncoc1C1CCCO1)=O c1(C(=O)NC2CCCN(C(c3ccc(C4CC4)s3)=O)CC2)cnc2ncccn12 C(=O)(CCC1=NNC(=O)CC1)NC1(CC)CCCN(C(=O)C(C)=CC(C)(C)C)C1 C1(C(=O)NCCC2(OCC)CCC2)C=CCN1C(=O)C(C)CC1CCCO1 c1(OC(C)C)ccc(C(N2CCC(C)C2CNC(=O)COCCC(C)C)=O)nc1 N1(C(c2c(C(C)C)scn2)=O)CC(N(C)C(C2CCCCCC2)=O)C(F)C1 Cc1cc(C(=O)NC2(CNC(=O)CC(C)c3cccnc3)CC2)cnn1 O=S(=O)(c1cc(F)c(F)cc1F)N1CCCC(O)C1c1ccc(F)cc1 c1(C(=O)NC2(CCOC)CCN(C(=O)C=C(C)C3CC3)C2)csc(S(C)(=O)=O)c1 c1(C(=O)NCC(CC)(C)NC(c2ccc(C(C)C)cc2)=O)cnn2ccccc12 C1(NC(c2cccc(Cl)c2F)=O)CS(=O)(=O)CC1NC(=O)C1=C(Cl)CCC1 N1(C(C(=O)NCC#C)C)CCC(C)C(NC(c2ccnc(F)c2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CC2CC(NC(c3nncc(C)c3)=O)C2C1 c1(OC)cc(CC(N2CCC(C(=O)NCC3(c4cccs4)CC3)CC2)=O)ccn1 CC1=C(C(=O)NC2CC(NC(C3(C)CC4CCC3C4)=O)C2)C(C)(C)CCC1 c1(C(C)C(=O)NCCN(C(=O)C=CC2CCCC2)C2CC2)ccc(C(F)(F)F)cc1 c1(C(N2CC(F)CC(NC(c3c(CC)cc[nH]3)=O)C2)=O)c(OC)ccc(Cl)c1C CC12CCCC(C(=O)NC3CCC(CNC(c4ccns4)=O)C3)(CO1)C2 C1(C(=O)NC(C)CCCNC(=O)CC2CCC2(F)F)(OC)CCC(F)(F)CC1 C(c1csc(Br)c1)=CC(N1CC(N(C(C2C(OCC)C2)=O)C)C1)=O c1(CCC)ccc(C(=O)NC(CN(C(=O)CSCC(C)C)CC)CC)cc1 N1(C(CC(CN(C)C)O)=O)C(CNC(=O)CC=C(Cl)Cl)CC2COCC12 Cc1nccnc1C(C)NC(C1(NC(=O)CCc2ncnn2C)CC1(C)C)=O c1(OC)cccc(C(=O)N(C2CN(C(c3cccc(N)c3)=O)CC2O)C)c1C N1(C(c2ccc(C#C)nc2)C(=O)NC2CCC2)CCN(C)C(=O)C1CC c1(-n2c(C(F)C(F)(F)F)nc(C)n2)ccc(F)c(Cl)c1 c1(OC)cc2c(cn1)NC2=O.N1(C(C2CC(O)C2)=O)CCCC(C)(O)C1 N1(C(=O)CNc2ccccn2)CCN(C(c2ccc(Cl)s2)=O)CC(O)C1 Cc1ccc(CN(C)C(C2C3CC2N(C(c2cnc(C)c(C)c2)=O)C3)=O)cc1Cl N1(C(c2ccc(C#N)s2)=O)CC2CCCN(C(c3csc4cncn34)=O)C2C1 c1(C(N2CC(C(=O)NCCNC(CS(N)(=O)=O)=O)C2)=O)ccc2[nH]ccc2c1F C=CCCCC(=O)NCC1CC1Cc1ccccc1.c12ccnc(c1)C(=O)NC2 c1(NC)cc(-c2cncnc2C(=O)OCc2ccccc2)cc(F)c1 n1(CC(=O)NCC2OCC(CNC(C)=O)C2)nc(C)n(C)c1=O C1(NC(C2CC(=O)N(O)C2)=O)CN(C(c2cc[nH]n2)=O)CC2(CCC2)C1 N1(C(c2n(C=C)ncc2)=O)CC2CCN(C(C3SCCC3C)=O)CCC2C1 N1(C(CCC=CC)=O)CCN(C(=O)Cc2ccc(O)c(C)c2)CC1CCC Cc1n[nH]c(C)c1CC(N1CC2C(NC(c3cc(C4CC4)on3)=O)C2C1)=O c1(C(=O)NCCCC(C)NC(C=CC)=O)ccc(C(=O)OCC)c2[nH]ncc12 C1(NC(c2ccc(NC)cc2)=O)CN(C(C2CC2(C)C)=O)C2(CCCC2)C1 c1(C(N2CCC(CC(C)NC(C(C(C)O)C)=O)CC2)=O)ccc2ocnc2c1 c1(C=O)ccccc1P(C)(C)=O.C1(C(N(CCCC)C)=O)CC2(CC2)C1 c1(C(=O)NCCCCNC(c2ccc(C(C)=O)[nH]2)=O)ccc(OC(F)F)cn1 C1(C(N(CCC(=O)OC)C)=O)CCCCN(C(=O)C(F)CC2CCOC2)C1 c1(C(=O)NC2C3CCN(C(c4n(C=C)nnc4)=O)CC32)c[nH]c2ccncc12 C1(C(N(CCC(=O)NC2CCN(CC3CC3)C2)C2CC2)=O)CN2CCC1CC2 c1(C(=O)NCc2cc(C(=O)NC(CC)C(C)O)n[nH]2)cccc(F)n1 C1(C(C)CO)CCCCN1C(=O)CC1CCN(C(C2CCCCO2)=O)C1 CC1CC(NC(=O)C=CCN(C)C)CN1C(c1cc(O)ncn1)=O Cc1ncnc2c1CC(C(=O)NCCC1(O)CN(C(=O)C3=COCC3)C1)CC2 C(=O)(C(C)(C)CO)N1CC(O)(CCNC(C2C(C)C2(F)F)=O)C1 C#Cc1cnc(C(=O)N(C2CN(C(c3cc(CCC)on3)=O)CC2O)C)c(C)c1 N1(C(c2ccc(CC)o2)=O)CC(C)CN(C(c2cc[n+]([O-])cc2)=O)CC1C N1(Cc2ccc(CC)cc2O)CC(NC(c2conc2C)=O)CC(F)(F)C1 CN1CCC(=CC(=O)NCC23CC2CN(C(c2cncc(O)c2)=O)C3)CC1 c1(C(C)OC(=O)C=Cc2cccc(-c3ccc(Cl)cc3)c2)ccc2c(c1)CCC2 c1(CC(=O)NCC2C(NC(C(C)N(C3CCCC3)C)=O)C2)ccc(F)cc1Cl C1(CNC(C=C(C)C(C)C)=O)CN(C(=O)CCC2CCCOC2)CC1C(N)=O C#CC1(C(N2CCC(CC(=O)N(C)CCc3ncon3)CC2)=O)CCCC1 C12(CNC(c3cnc(CC)s3)=O)CCCC1N(C(=O)CCn1cncn1)CCC2 N1(C(COC(C)C)=O)CC2(C1)OC1(CNC(c3ccccc3)=O)CC2(C(N)=O)C1 C1(CC)CN(C(C2(CO)CC2)=O)CCN1C(c1cc(Br)ccc1N)=O N1(C(C(C(C)C)n2ccnc2)=O)CC2CC1CN2C(c1ccc(Br)o1)=O Cc1coc(C(=O)N(C)CCNC(C2(NC(=O)Oc3ccccc3)COC2)=O)c1C CN1CCCC(O)(CC(N2CCCCC2CCN(C)C(C2(F)CCCC2)=O)=O)C1 C1(C(NOC(CC)C2CCC2)=O)CC(F)(F)CN1C(C1CCOC1C1CC1)=O C=C(Br)CC(C)(C)C(=O)N(C)CCOCCNC(c1ccc(COC)o1)=O c1(C(=O)NC(C2CCN(C(c3c[nH]nc3Br)=O)C2)C)cccn2ccnc12 c1(OC)ccc(C=CC(=O)NCCCCN(C(=O)C(C)C2CCCO2)C)cc1 C1(C(=O)OC)CN(C(=O)C(C)Oc2ccc(Cl)cc2)CC(C)(C)S1(=O)=O C12(F)CCN(CC1)C2.CC1(C)C(NC(c2cnn(CCF)c2)=O)C1C(F)F c1(C2C(C)C2)ccc(C=CCN2CCC(N(CCC(F)(F)F)C(=O)C3CC3)C2)o1 C1(NC(C2(OC)CC2)=O)CCCCC1N(C(=O)COc1cccc(F)c1)C c1(C(=O)NCCCC(C)NC(=O)CC(C)c2cnn(C)c2)nnc(O)cc1O N1(C(CCCC#CC)=O)CCC2CC2(NC(c2ccc3cnoc3c2)=O)CC1 N1(C(C=CCCC)=O)CCC2(CC1)CC2NC(=O)Cc1cc(Cl)cnc1C c1(C(=O)NC2CC(C)CN(C(c3ccc(Cl)[nH]3)=O)C2)cccc2c1OCCN2 C1(C(N2CCCC(NC(=O)Cc3ccn(C(F)F)n3)C2)=O)CC(C2CC2)=NO1 C(c1cc(Br)ccc1OC)=CC(N1CCC(NC(CCCOCC)=O)C1)=O c1(OC)ccc2[nH]nc(NC(C3(CNC(c4cc(Br)cnc4Br)=O)CC3)=O)c2c1 c1(OC)cncc(C(=O)NCCC(C)NC(c2cc(Cl)ccc2Cl)=O)c1C C(=O)(CC(F)(F)C(C)C)NC1CN(C(CCc2cnc(C)s2)=O)C(C)CC1 C#Cc1cccc(OCC(N2CCC(F)(CNC(=O)Cc3nncs3)CC2)=O)c1 C1(C(=O)NC(C(C)C)CCNC(C2CC2(C)C)=O)CN2CC3CC2(CO1)C3 c1(N2CCCC(Oc3ccc(OC)cc3)C2)nc(Br)cn(C)c1=O C1(CC(=O)NC(CN(C(Cc2ccc(SC)s2)=O)CC)C)CCc2c(ncn2C)C1 N1(C(C(C)O)=O)Cc2nccn2CC(NC(=O)COCC2CCCO2)C1 C1(C(=O)NCC=CCC(=O)NCCCC2(C)CC2)COCOC1 N1(C(C2CC(N(C)C)C2)=O)CC(=O)NCC1C(N1CCC(C)(CCO)C1)=O C12(CC)CN(C(=O)C(C)C3CC3)C(CNC(=O)C(C)Cc3ccccc3)(C1)C2 CN=c1ccc(C(N2CSCC2C(=O)NC2C3CCC2CC3)=O)c[nH]1 C1(N(CCOn2cccn2)CC)CCN(CC(C)C)CC1 N1(C(C#C)=O)CCCC2C1CCN2Cc1cc(OC(F)(F)F)cc(F)c1 CC(C)CC(=O)N(CC(O)CN(C(=O)CN(CC(C)(C)C)C)C)C c1(C(=O)NCC(=O)NC(C(=O)N(C)CCN(C(=O)CO)C)C)cccnc1S S(=O)(=O)(c1cccc(C(=O)Nc2ccccc2[N+](=O)[O-])c1)N(C(C)(C)CO)C C1(NC(CC(C)CN(C)C)=O)CC(F)CN(C(c2ccc(N)cn2)=O)C1 N1(C(COC2(C)CCCC2)=O)CC(=O)NCC1C(=O)NCCC1CCC1 N1(C(CCCOC(C)=O)=O)CC2(CCCC2)C1C(=O)NC1CCOCC1C c1(CCC)ccc(C(=O)NC2CN(C(=O)C(C#N)C3CC3)CC2F)cc1[N+](=O)[O-] CC(C)CC(CC(=O)NC1(CCCNC(c2cncnc2)=O)CC1)CC(N)=O CCC(C)C(O)C(C)C(=O)N(C)CC=CC(=O)NCC1(N(C)C)CCC1 C(C(C)(C)C1=CCOCC1)NC(=O)Nc1cc(C)n(C)c1C c1(CC(=O)N(C2CCN(C(C3CCOC3C)=O)C2)CC)ccc(C(C)C)cc1 C1(COC)CCCN1C(=O)COC1CC(NC(=O)C=Cc2ccsc2)C1 N1(C(C2C(C)OCCO2)=O)CCC2CN(C(C3CCSCC3)=O)CC2CC1 C1(CC)CC(C(N2CCN(C(C3CC(C)(C)CN3C)=O)C(CO)C2)=O)CC(=O)N1 C1(C(=O)NC2CC(CCC(=O)NCC3(C)CCCO3)C2)CC2(CCC2O)C1 c1(C(=O)NC2C(C(N3CCC(CC#C)CC3)=O)CCC2)cccc(C#N)c1C CC(C(=O)NC1C2CCCC12)(C1CCC1)NC(C1CC(=O)C1)=O C1(N(C(C2CCC(F)(F)C2)=O)CC)CCCN(C(=O)CCN2CCCCC2)C1 c1(C(=O)NC(CC2CN(C(COCC#C)=O)C2)C)cnn2cccnc12 N1(C(=O)OC)CCCN(C(=O)C(=O)Nc2c(C)cccc2C)CC1C(=O)OC C1(C)(CC)CC(NC(=O)Cc2ccncc2Cl)CN1C(=O)CN1CCCC1 c1(C(=O)OC)cccc(C(N2CCOC(CNC(C3CC(C)(C)CO3)=O)C2)=O)c1 Cc1cc(CC(=O)NCc2csc(C(=O)NC(c3ccccn3)CO)c2)n(C)n1 C(=O)(CC(C)(C)C(F)F)Nc1c(C)cc(NC(c2cnc[nH]2)=O)cc1 c1(C(N2CCC(N(C(C=CC)=O)C)C(C)C2)=O)ccc2c(c1)CCN2C N1(C(C2CCCN(C(c3cc(OC)c(C)cc3)=O)C2)=O)CCCC2(CCNC2)C1 C12(C(N)=O)CCCC1(C(=O)NC1CCN(C(=O)C(F)n3ccnc3)CC1)C2 N1(C(C=C(C)Cl)=O)CCN(CCN(C)C(c2ccnc(-c3ccco3)c2)=O)CC1 Cc1cc(Br)cc(F)c1NC(=O)C(N1CC2CCNC2(C(F)(F)F)C1)=O C1(NC(C(C)(C2CCC2)NC(=O)C=Cc2cocn2)=O)CCCCC1O N1(N2CC(n3cc(C4(C)CCCO4)nn3)C2)CCC2(CC1)CC(O)CCO2 C1(CNC(c2cccc(OC(CC)C)c2)=O)N(C(=O)CSC(F)F)CCC1(C)C N1(C(C(CCC)NC(C2(C(=O)OC)CC2)=O)=O)CCN(C)CC1CCO C12(CN(C(=O)C(C)CN(C(=O)Cc3cnnn3C)C)CC)CCC(CC1)C2 C1(C(=O)NC(C(=O)NCCC2(COC)CC2)C2CCCO2)OCCC1(C)C C(=O)(C1CCCn2c(C)cnc21)N1CCC(CCNC(C(CC)O)=O)CC1 N1(C(C2(CC(C)C)CCC2)=O)CC2(C(=O)NCC3CCCS3)CC1CO2 N1(C(C=C(CC)CC)=O)CC(NC(C2CC(n3ccnc3)C2)=O)CC(F)(F)C1 Cc1cc(C(=O)NCCCOCCC(=O)NC2CCOC2(C)C)nnc1O c1(C(N2CC(O)(CCNC(=O)CCCC(F)(F)F)C2)=O)ccc2c(n1)CCC2=O CC(C)C(C)C(C)CC(=O)N1CCC(NC(=O)COCc2ccccn2)C1(C)C O=C(C1=C(Cl)CCC1)NC1CC(NC(C2(c3ccccc3)CC3(CC3)C2)=O)C1 C12(C(N3CC(C(C)C)OCCC3)=O)COCC1CN(C(=O)CC1CSCCO1)C2 C1(C)(CC)CC(NC(c2ocnc2C2CC2)=O)CN1C(=O)Cn1cccnc1=O C(C)(C)(C(=O)NCC(CNC(=O)CCCn1c(C)cnc1O)OC)OCCC C(CC1CCC1)(C(=O)N1CCCO1)NC(CC1N(C)CC=CC1)=O N1(C(Cc2c(C)nc(S)s2)=O)CCN(C)CC1CNC(=O)C(C)NC(N)=O c1(C(=O)NC23CC(CNC(C4C(C)CC4C)=O)(OC2)C3)cncc2ncn(C)c12 C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NC(C)CNC(C1CCCC12CC2)=O c1(CC(=O)N(CCC)CCNC(=O)CC2C=NN(C)C2=O)cccc2ccoc12 c1(C(N2CCC(NC(C(C)NC(C)=O)=O)C2)=O)c(Cl)ccc(C)c1O N1(C(C(C)c2cccs2)=O)CCCC(CCNC(=O)CSc2ccncc2)C1 C(CC(C)(C)C(=O)NCC1(F)CCC(NC(C2CCC(=O)NC2)=O)C1)OC c1cc2nnnn2c2c1C1NC(=N2)N(C)C(CC)CCC2CCN(CC1)C2 c1(C(N2C(CO)CC(NC(C3C(OC)C3)=O)C2)=O)cc2ccncc2s1 CS(=O)(=O)c1ccc(C(N2CCCC3(NC(c4cscn4)=O)CC3C2)=O)o1 C1(OC)CCCC(Nc2cccc(-c3cncn3C)n2)C1 c1(NC(C2(C)CC2(F)F)=O)cnc2sc(-c3ccccc3)cn12 CC(CC(=O)NC1(CO)CCC1)C(C)(C)NC(c1cnn(C)c1)=O n1(CC)nnc(C(=O)N(CC(C)NC(C2CC2c2cnn(C)c2)=O)C)c1C C(C(O)C(F)F)NC(CC1(N(C)C(c2cc(COC)on2)=O)CC1)=O n1(CC(=O)NCCCC(C)NC(COCC(=O)OC)=O)ccc2cc(F)ccc12 C1(NC(C=CCCC=C(C)C)=O)CN(C(C2(C)CC(F)C2)=O)CC2(CCC2)C1 c1(C(=O)OC)csc(CNCc2cn(-c3ccn(C)n3)cn2)n1 N1(C(C2(CC#C)CCCO2)=O)C2CCC1CN(C(C1CCC(=O)N(C)C1)=O)C2 C1(N(C(C(n2cc(C(F)(F)F)nn2)C)=O)C(C)(C)C)CCOC(C(C)(C)C)C1 C(=O)(C(C)(O)CC(F)F)NCC1(CNC(C(n2cc(C)nc2)(C)C)=O)CCC1 CCC(CC(F)F)C(=O)N1CCCC(CN(c2ncc3ncnc-3[nH]2)C)C1 C1(CC(N2CCC(CC)C2)=O)CN(C(C2(C(=O)OC)CC2)=O)CCC12CCC2 c1(NCCOCCNC(=O)CC2(C(F)(F)F)CC2)ncc2ccccc2n1 C12(CNC(=O)COCC(F)(F)F)CCCCC1CN(C(c1cocn1)=O)C2 C1(C2C(c3c(C)cco3)C2)CCC2(CC1)CN(Cc1cnc(C3CC3)o1)C2 N1(C(C2(CC=C)CN(C(=O)CC3(C#N)CC3)C2)=O)CCC(C)(C)C1C c1(C(=O)OC)ccc(O)nc1NCC1(NC(c2cc(=O)n(C)cn2)=O)COC1 N1(C(C(=O)NCCCCCC)C2CC2(C)Br)CCC(O)(CCC)CC1 N1(C(c2nccc(CC)c2)=O)CCC2(CC1)CC(NC(=O)CNC(C)=O)CO2 c1(CNc2cncc(C(=O)NCCn3cc(COC)cn3)c2)c(I)ccnc1Cl C(=O)(C#CC(C)(C)O)NC(CC(C)C)CNC(=O)Cc1cn[nH]c1 C(=O)(CCCCC(=O)N1CCCC1CCNC(=O)Cc1conc1C)OC Cc1cc(C)c(C(N2CCN(C(c3cc(Cl)c[nH]3)=O)C(C(C)(C)C)C2)=O)cc1C CC1(C(N2CC(NC(C3CC(OC(F)(F)F)C3)=O)C(O)C2)=O)CC=CCC1 c12cnc(s1)C2.C(C(C)(C)C)C1(C(=O)NC(C2C(C(=O)OCC)C2)C)CC1 S(=O)(=O)(c1ccc2cc(Cl)sc2c1)N1CCN(c2cc(C)nc(C)n2)CC1 Cc1cc(C(N2CC(NC(=O)CN3CCCNC3=O)CCC2C)=O)cc(N)c1O CN1N=C(CC(=O)N2CC(NC(=O)CC3CCS(=O)(=O)C3)CC3(CC3)C2)CC1=O C1(CN(C)C)NC(=O)N(CC(C)(C)CN2CCOCC2)C1=O CC1COCC(CC(=O)NCCCN(CC(=O)Nc2ccccc2Cl)CC2CC2)O1 CCCS(=O)(=O)C(C)C(=O)NC1(C2CN(C(=O)C=Cc3ccc(F)nc3)C2)CC1 N1(C(C(C)OCCCCCC)=O)Cc2[nH]nc(C(=O)N(C(C)CO)C)c2C1 N1(C(C(CC)OC)=O)CCC(COC)(NC(C2CCC(F)CC2)=O)CC1 C(CC(=O)NC1(C)CCN(C(C2(c3cccc(Cl)n3)CC2)=O)C1)(C(F)(F)F)OC c1(NC(C2COC3CN(C(CCC=C)=O)CC32)=O)ccc2c(c1)OCC(=O)N2 CC(C)C(CC(=O)NCCS(C)=O)NC(=O)CCCn1cccn1 n1(CC(N2CCC(NC(C)C)CC2)=O)cnc2c1CCCC2 C1(NC(CCn2cc(C)nc2)=O)CC(C2CCCC2)C1 N1(C(=O)CCc2nccs2)CC2CN(C(C3(O)CCC3)=O)CC2C1 N(C=CC(=O)C(F)(F)F)C(=O)CCCCCl.Cn1cc2nc1C(=O)N2 c1(C(=O)NCCCN(C(c2nccc(C(F)F)n2)=O)CC)cn(C)[nH]c1=N C1(C(=O)NCC(C)NC(C(C2CCOCC2)OCC)=O)CC(=O)NC(=O)N1 n1(CC=C)cc(C(=O)NCC2CC(O)(CNC(c3cc(C)sn3)=O)C2)cn1 c1(OCC=C)ccccc1C(=O)NC(CO)C(C)NC(C1CCCC1CC)=O C1(C)C(C2CC2)CCN1c1ccccn1.c1(O)ccc(CCC(=O)NCCOC)cc1 C12(CC(=O)NCCCc3nnc(C)o3)CCC1CN(Cc1cc(Cl)ccc1Br)C2 Cc1cccc(F)c1C(=O)NC1CCN(C(c2occc2Br)=O)C1C CC1C(C)N(C(c2cc(Cl)ns2)=O)CCN1C(c1noc2ncccc12)=O C1(n2c(C(n3ccnc3)CC)nc(-c3cccc(F)c3)n2)CCCCC1(C)C c1(CC(=O)NCCNC(=O)CCc2ncc[nH]2)cccnc1Br c12ccnc(c1)N1CCN(CC1)C2=O.c1(C(=O)NC2CC2)ccc(OCF)cc1 C12(CC(=O)NCC3CCCN3C(=O)C(C3CCCCC3)O)CCC(CC1)OC2 C(=O)(CCCCC(N)=O)NCC(COC)NC(c1[nH]cc(CC)n1)=O C1(NC(c2cc(C)sn2)=O)CC2CCC1C(NC(=O)CC1CCCC3(CC3)C1)C2 C12(NCc3[nH]nc(COC)n3)CCCCC1N(C(c1cc(F)ccc1F)=O)CC2 Cc1cccc(C(N2CCC(N(C)C(C34CC(C)C3C4)=O)C2)=O)c1F C1(C(=O)NCC2(O)CN(C)C2)(OC)CN(C(=O)C(c2ccccc2)O)C1 c1(C(C)C(N2CCC(Cc3cn(CN4CCCC4)nn3)C2)=O)ccc(C#N)cc1 C#Cc1cnn(CC(N2CCOC(C(=O)NCCC(C)CO)C2)=O)c1 c1(C(=O)NCCC2(C)CCN(C(COCCC#C)=O)C2)cc(OC)ccc1C c1(C(=O)NC2C(CC)CN(C(=O)CCCC(C)C)CC2)cn2ncnc2nc1C N1(C(CCCCC)=O)CCC(C=CC(=O)NC2C(O)CC2O)CC1 C1(N(C(CN2CCC(C)C2)=O)C)CN(C(=O)Cc2ccc(F)cc2F)CC12CC2 Cc1cc(Br)c(CC(=O)NC2CCC(CCNC(c3cnc[nH]3)=O)C2)s1 C1(C(=O)NC(CC)C2CC2)CC(C)CCN1C(=O)C(O)CSC c1(OC)ccc2[nH]c(C(=O)NCC3CN(C(=O)CCC=C(C)C)CCO3)cc2c1 C(=O)(CC1=CCN(C(=O)CC=CC(C)(C)C)CC1)N1C(C)CC(CO)C1 c1(CC)cc(C(=O)NC(C)CN(C(=O)CSC2CCOC2=O)CC)nn1C CC1(C(=O)NC2CC(NC(=O)Cc3cncnc3)C2)CCC2(CC1)CC2 N1(C(=O)CCn2cccn2)CC2CC(C(N3CCCC(F)(CO)C3)=O)C(C2)C1 Cc1cc(F)c(C(N2CC(NCc3ncnn3CC(C)C)C(O)C2)=O)cc1F C1(CN(C(=O)C(C)(C)F)C)CCCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 c1(C(=O)NC(CCCCNC(C(F)=C(C)C)=O)C)cccc(Br)c1[N+](=O)[O-] c1(CNC(C(C)OCC=C)=O)ccc(C(=O)NCc2cc(C)sc2C)cc1 c1(C(c2cn(CC(=C)CC)nn2)NC(=O)N(CC(=O)OC)C)ccc(F)cc1C C(CCCCC(=O)NCCCNC)NC(c1c(CCC)n[nH]c1)=O c1(C(C(=O)NCCCN(C(C=CCC)=O)CC)OCC)ccccc1 c1(C(=O)NCC(C2CCCC2)NC(C(C)=C2CC2)=O)nc(CC2CC2)oc1C C1(O)(C(=O)NCC2CCN(C(CC(C(=C)C)OCC)=O)C2)CCCC(C)(C)C1 c1(C(=O)NCCn2cc(CNC(C3(CC)CCC3)=O)nn2)cc(C)cnc1F c1(N(CC(=O)NC2CC(n3ccnn3)C2)C)ccc(Cl)cc1 c1(C(=O)NCC2(NC(c3n[nH]c(C)c3Br)=O)CC2)ncnc2sccc12 C1(c2cccs2)(C(N(CCN(C(CNS(CC)(=O)=O)=O)C)C)=O)CC(F)(F)C1 N1(C(c2cnc(C)s2)=O)CCCC(N(C(=O)C2=CCSC2)C)C1 Cc1ccc(C)c(C(=O)NCC2CN(C(C3CCOC3)=O)CC23CC3)c1O c1(OC)ccc(C)cc1-n1cc(C2CN(C(c3cnc(C)o3)=O)CC2(F)F)nn1 N1(n2cc(C3OCCN(C(c4cc(F)ccc4F)=O)C3)nn2)CCOC2CSCC12 N1(C(C2(CC)CCN(C(=O)CCC(CF)CF)CC2)=O)CCC2(C1)CC2(F)F CC1(C)CCC(CCNC(=O)C(c2ccco2)NC(=O)C(=O)N(C)C)O1 C1(NC(c2c(C)occ2)=O)CCN(C(c2c(Br)ncn2C)=O)CC1 C1(C(N2C(CNC(=O)CN3CCCCCC3)COCC2)=O)SC2C=CC1CC2 N1(C(c2cc(CC)on2)=O)CCC(NC(=O)C(c2c(C)n[nH]c2C)C)C(F)C1 CN=c1[nH]c(=NCC2CCc3nccn3C2)[nH]c(=NC(C)c2ccnc(Cl)c2)[nH]1 Cc1ccc(N(C)C(C2C3CN(C(c4ccns4)=O)CC23)=O)c(C)c1 N1(C(C(CCC)(C)C)=O)CCCC(C2CCN(C(C3(CO)CCCC3)=O)CC2)C1 c1(C(=O)NC2C(CC)CN(C(c3nn(C)nc3C)=O)CC2)ccc2nnnn2c1 C#Cc1cc(C(=O)NCC2CCCN2C(C2CCCN2CCC)=O)ccc1Cl C1(C(=O)NC(c2cc(F)ccc2F)C)CCCN(C(=O)Cn2ccnc2)CC1 C1(C(=O)NCCC(C)CCN(C)C)NCCN(C(=O)OC(C)(C)C)C1=O CON1CCC(CC(=O)NC2CC(CC(=O)NCCc3nc(C)no3)C2)CC1 Cc1cc(CCC(=O)NC2CN(C(=O)CN(c3ccc(Cl)cc3)C)C2)nn1C C1(O)(C(CNC(C(C)SC(C)C)=O)(C)C)CN(C(c2ccc(C(C)(C)C)[nH]2)=O)C1 CCC(F)(F)CC(=O)NCc1occc1C(=O)N(C)Cc1cncnc1 c1(CC)ccc(C(=O)NCC(C)NC(c2nc(Cl)oc2C)=O)cc1Cl c1(C(=O)NC(CNC(=O)Cc2cn[nH]c2)CC(F)(F)F)c(F)cc(F)cc1F c1(CNC(COC)=O)ccc(OC(F)(F)F)c(C)c1.C12CCCC(C1)NC2=O CC(CS(C)(=O)=O)C(=O)N1CC2CC2(CNC(c2ccnc(C(F)(F)F)c2)=O)C1 N1(C(C(C2CC(NC(c3cnn(C(C)C)n3)=O)C2)F)=O)CCCC(N=[N+]=[N-])C1 C1(C(=O)NCc2ncc(OC)nc2)CC(=O)OC12CCCCC2 c1(C(N2CCCC(Cn3cc(C=CC)nn3)C2)=O)ccc(C)cc1C N1(C(C(C=C)(F)F)=O)CCCCC1C1CCCN1c1ccnc(C(C)CC)n1 C1(C(N2CC(CCNC(C=C(C)Cl)=O)OC(C)C2)=O)CC2C=CC1C21CC1 C1(CNC(COC(C)=O)=O)CC2CCC1N(C(c1cn(C(C)C)nc1C)=O)C2 CC1CCN(C(c2ccc(CNC(=O)C=CCF)nc2)=O)CCO1 c1(C(NOCCC#C)=O)coc(CNC(C2CCCC2OC)=O)c1 C1(n2cc(-c3scc(C)n3)nn2)CCC(NCCC(=O)NC(=O)C2CC2)CC1 C1(NC(C(CC)NC(N)=O)=O)CCN(C(C2CCC=CCCC2)=O)CC12CCC2 Cc1ccc(C)c(-c2nc(Cc3cccs3)nn2Cc2ccc(C)o2)n1 N1(C(CC2CN(C(CSCCOC)=O)C2)=O)CCOC2(CCN(C)C2)C1 c1(CC(=O)OCC)ccc(OC)cc1NC(=O)C(c1ccc(Cl)nc1)N N1(C(C)=O)CC(NC(=O)Nc2cnc(-c3ccccc3)nc2C)CC(O)C1 c1(OC)cc(CN2CCOCC2C(=O)Nc2nc(Br)ccc2OC)cc(Cl)c1O C(CCC(C)C)(C(=O)NCc1oc(C)nc1C)NC(c1cc(C)nc(C)c1)=O C=CCC(CC(C)C)C(=O)N1CCN(C(c2ccc(=O)n(C)c2)=O)C(CO)C1 C1(CCOC)CN(C(c2ccc(C(C)C)o2)=O)CCN1C(=O)CN1CCCCC1 c1(NC(c2c(C)n[nH]c2C)=O)cnc(Cl)cc1C(N1C2CCC1COC2)=O CC(C)CC(C)C(=O)NCC1CCN(C(=O)C#CC(C)(C)C)C1 Cc1cnc(C(=O)N(CC(C)(C)CNC(=O)CNc2nccs2)C)cc1C c1(C(=O)NCCCCNC(C2(C(=O)NC)CCC2)=O)cccc2nonc12 Cc1cc(C(=O)NCC2(CNC(C3CCC(C)S3)=O)CC2)cc(N)c1Cl c1(C(=O)NC2C(C)CN(C(c3c[nH]cc3Br)=O)C2)cc2ccc(F)cc2[nH]1 C=CC(CCC)CC(=O)N1CCCC(C(=O)NCC(=O)NC2CC2)CC1 C=CC(C)(C)CC(=O)NC(C1CCCCC1)C(N1CC2(CCOC2)C1)=O C(N=c1[nH]c(=NCCN2CCC(C)CC2)[nH]c2c1CCC2)C1CCC(CC)O1 c1(C(=O)NCCC(CNC(c2c(C)ncn2C)=O)O)ccc2c(c1)NC(=O)CO2 N1(C(CN(C(C)=O)C)=O)CCC(C)(c2cn(C(C3CCCO3)C3CC3)nn2)CC1 c1(CNC(=O)C(=O)NC(C2CCCCC2)C2CC2)nc(Br)c(Br)cc1Cl Cc1cnc(C(=O)NC(C23CCC(C(=O)NC4CS(=O)(=O)C4)(CC2)C3)=O)cc1F CC1CN2CCN1C(C(N1CC(OCCNC(C3CCCCNC3=O)=O)C1)=O)C2 C1(C(=O)NC(CNC(C2(O)CCCC2)=O)C2CC2)CSc2ccccc2O1 S(=O)(=O)(c1ccc(C)c(Cl)c1)NCC(=O)OC(=O)CC1CCCCN(CC)C1 C1(NC(=O)C(O)Cn2cncn2)CC2CC(NC(C3C4CCCCC34)=O)C2C1 C1(CNC(CCc2cnc(C)o2)=O)CCN(C(c2c(C)nn(C)c2F)=O)CC1C C1(N(C(=O)C2=NOCC2)CC)CCCN(C(c2ccc(C(C)C)o2)=O)CC1 C(C(C)(CC(C)C)NC(c1coc(Br)n1)=O)NC(c1c(CC)n(CC)nc1)=O N1(C(Cc2cn(CC)nc2C)=O)CCN(C(=O)COc2ccsn2)C(CO)C1 c1(C(=O)NCCC2(NC(C3C(CCOC)C3)=O)CC2)cc(Cl)cs1 N1(C(c2c(NC)snc2C)=O)CCC(C)(C)C(NC(c2ccc(N)cc2F)=O)C1 n1(CC(=O)NCCn2cc(-c3ccccc3)nn2)nc(-c2cccs2)ccc1=O CC(C)(C)CC(F)C(=O)NCCCN(C1CCCC1)C(C1C(C(F)F)C1(C)C)=O c1(OC)ccc(C(C)CC(=O)NCC(C)NC(=O)CCc2cccnc2)cc1 CC(C)C1=NOC(C(N2CCCCC2CC(=O)N(C2CCCCCC2)CCO)=O)C1 C1(NC(COCC=C)=O)COC2CN(C(c3nc(Cl)ccc3N)=O)CC12 c1(C(N(CC(CNC(COCCCC)=O)C)C)=O)cnc2ccc(C)cn12 C(=O)(C(C(C)(C)C)NC(=O)CC1COCC(C)O1)NC(C(C)SC)C O=C(CCc1ccon1)NC1CC1NC(C1(C(N)=O)CC1)=O C1(C(c2sc3ncc(NC(C(=O)N(C)C4CC4)=O)n3c2)=O)COC2(CCNCC2)C1 c1(C(=O)NC2C(NC(C3(COC)CCCC3)=O)CC2)cc2ccccc2c(O)n1 N1(C(C2CC(CC)(CC)C2)=O)CCC(O)(C(C)NC(=O)CCc2ncc[nH]2)CC1 c1(C(=O)NCCCN(C(=O)C(F)n2ccnc2)CC)nnsc1C(F)F c1(C(=O)NC2CCC(F)(CNC(CCOCC)=O)C2)cccc(SC)c1[N+](=O)[O-] C#Cc1ccc(CC(=O)NCCCCC=C)cc1.N12CCC(CF)(C1)C2=O N1(C(CNC(=O)OC)=O)CCCN(C(C2CCC(C(C)C)NC2=O)=O)CC1 C(CC(C)C(=O)N1CC(O)CC1CNC(=O)CCCn1nc(C)nc1C)OC N1(C(CCNC(C)=O)=O)CCN(C(=O)CC2COCCO2)CC(C)C1 Nc1ccc(C(=O)NCC(CNC(C2CC3C(C2)C3(F)F)=O)CO)nc1F c1(SCC)cccnc1C(N1CCC(NC(=O)Cn2nnc(C3CC3)n2)CC1)=O C(=O)(C(O)CC(N)=O)N1C(C)C(C(=O)NCCCN(C)C2CC2)CC1 N1(C(=O)Cc2cnns2)CCC(c2cn(CCOCCO)nn2)C1 C1(NC(C(C)C2CCCC2)=O)C=CCN(C(=O)CCC(=O)N(C)C)C1 N1(C(c2c(OC)ccnc2F)=O)CCCN(C(=O)C(O)C(F)(F)F)CCC1 C1(N(C(C2C(=C)C2)=O)C)CCN(C(=O)COc2cc(F)cc(F)c2)CC12CC2 C1(C(=O)NC(C)CCCNC(C23CC(C2)C(C)O3)=O)CCC2CCC(=O)N12 C1(C(=O)NC2C=CCN(C(C3OCCO3)=O)C2)CC12CC(F)(F)C2 N#Cc1cc(NC(C2(F)CN(Cc3cnc(Cl)nc3)C2)=O)c(Br)cc1F c1(C(=O)NC(C2(C)N(C(C(CC)COC(C)=O)=O)CCC2)C)cc(O)nc(Cl)c1 C1(CC(=O)NCC(C)NC(N)=O)CCCC1NC(=O)Cc1ccnn1C N1(C(C2CC(=C)C2)=O)CC2(CCN(C(=O)C(CC)CCCC)CC2)CC1C C1(NC(CCC)=O)CC1C1CCN(C(c2c(F)ccc3c2OCO3)=O)CC1 c1(CN2CCC(C)(C(=O)N(CCCO)CCCO)C2)cc(Cl)nc(Cl)c1 c1(-c2ccc(CNC(c3c(C)occc3=O)=O)cc2)cnn2ccc(O)nc12 C#Cc1ccc(CC(=O)NC(C)C=CCNC(C2CC(C)(C)CCO2)=O)cc1 N1(C(C2(C)CC2(F)Cl)=O)CCC(F)(CNC(=O)Cn2ccc(C(F)(F)F)n2)CC1 Cc1sc(CC(F)(F)F)nc1C(=O)NCCCN(C(C1(O)CCOC1)=O)C1CC1 C=C(CNC(=O)C=CC(F)(F)F)CCNC(=O)CCC1CC1(C)C c1(C(=O)NCC2COCCN(C(C(C)OC)=O)C2)cc([N+](=O)[O-])cc(C)n1 N1(Cc2n[nH]cc2[N+](=O)[O-])CC2CC(N(C)Cc3ccn(C(C)C)n3)C1C2 C1(NC(c2nc(CN(C(CCOC)=O)C)oc2)=O)CC=C(C(C)C)CC1 CC1CC(C(N2CCC(F)(C(N)=O)C2)=O)CCN1C(C1CN(C(N)=O)C1)=O S(=O)(=O)(c1ccc(F)cc1)NCC(=O)N(CC(=O)NCC1CC(C)(F)C1)C C1(CNC(CS(CC)=O)=O)CC12CCN(C(=O)C(=O)N(C)C)CC2 C(=O)(CCCC(C)O)NC(CC(C)NC(c1nc(COCC)sc1)=O)C c1(C(=O)NCCN(C(=O)Cc2ccnn2C)CCC)ccccc1-n1cncn1 c1(C(=O)NC2C3CN(C(CCCSC)=O)CC2C3)cc2cc[nH]c(=O)c2s1 c1(N(C(C)CCNC(c2ccc3nonc3c2)=O)C)[nH]cnc2nc(Cl)cc1-2 C1(CCNC(C(C)=C2CC2)=O)CN(C(C)=O)CCO1 C1(c2n(Cc3c(SC)nccc3)nc(-c3ccoc3)n2)CN2CCCCC2CO1 C1(CNC(C=CC(CC)C)=O)CC(NC(=O)CCOCC(F)(F)C(F)F)CCO1 c1(CNC(C2CC2C(N2CC(Oc3ccc(F)cc3)C2)=O)=O)cc(F)ccc1Cl c1(CC(N(C=O)Cc2ccc(F)cc2)=O)cccc(Br)c1 C=CCC(CC(C)C)C(=O)NC1CCN(c2nccs2)CCC1CO C1(CNC(=O)CC(F)(F)F)CN(C(=O)CN2CCCCCC2)CC2CC12 c1(OC)cccc(CC(N2CCCC2c2c(OC)cccc2O)=O)c1Cl C1(CNC(CN(C)CC)=O)CCC(NC(=O)CC(C)OCc2ccccc2)C1 C#Cc1ccc(OC)c(C(=O)NCC2CC2CNC(C2(S(C)(=O)=O)CC2)=O)c1 Cc1ccc(F)cc1CNC(=O)C(C1(O)CN(C(=O)CC2CSC2)C1)F c1(C(N(C(C)C)C)=O)ccccc1C(=O)NCC1(CCNC(=O)C(C)O)CC1 C(C(=O)NCC1(CN(C)C(c2cncc(Cl)c2)=O)CC1)(C(C)C)OCC N1(C(C2CC(CC)OCC2)=O)CC2(CCN(C(=O)CSS(C)(=O)=O)CC2)C1 Cc1cnnc(O)c1C(N1CCCC1CN(C)C(C1CC(=O)NC(=O)C1)=O)=O c1(OCCCC)ccc(CN2CCC(C)(NC(c3snnc3C)=O)C2)cc1 c1(Sc2c(CNCC(C(C3CC3)OC)(F)F)cccc2)nnc2n1CCCCC2 C1(C(N2C(CNC(C3(C(C)(C)C)CCCC3)=O)CC2)=O)CCC2(CC2)C1 C1(C(C)C)(C(=O)NC2CC2NC(c2cn(C(F)F)cn2)=O)CNC(=O)C1 C(=O)(CC(O)C(C)C)N(CCN(C(C1CC=C(C)CC1)=O)C(C)C)C C1(CNC(C2N(CC)CCOC2)=O)CC(F)(F)CN1C(c1sccc1OC)=O CCC(CC)CCC(=O)N1CCCC(O)(CNC(=O)C(C)NC(=O)NC)CC1 C(=O)(CCCC(F)F)NCC=CCNC(c1nc(C)[nH]c1C(F)(F)F)=O C(C(C(=O)NCC1CC2(CC2)CN1C(=O)C(=O)NC(C)C)C(C)(C)C)OCC=C C1(CNC(=O)CC2CCOC2=O)CN(C(=O)COCC(F)(F)F)CC1(F)F CC1CC(NC(=O)C(CC2CC2)NC(C2CCCCCC2)=O)CCO1 O=C1CC(C(=O)NCCc2nccc(O)n2)N(C(C2CCCC(=O)N2)=O)C1 C1(C(N2CC(CCNC(C3CC(N(C)C)C3)=O)C2)=O)COc2ccccc2O1 C1(C(C)NC(C(C)OC)=O)CCN(CC(=O)Nc2ccc(F)cc2)CC1O C1(CC)CN(C(c2ccc(CC(N)=O)cc2)=O)CCC1NC(=O)C(COC)CC c1(NC(c2n(CC)ccn2)C)nc(N2CC3(CCC3)CC2CO)nc2sccc12 C1(OC)CN(C(=O)CCC2CCOCC2)CC1NC(C1CC2(CC2)CO1)=O C1(CC)CN(C(C)=O)C(CC)CN1CC(c1ccn(CC)n1)(C)C N(C(=NCN1CCCC1)NCC(C)(C)C(F)F)C(CN(c1ccsc1)CC)C N1(C(=O)OCC)CCC(NCCC(C)N(C)Cc2cn(CC(=O)N(C)C)nn2)C1 N1(C(C2CC(=C)C2)=O)CCCC(C(C)N(C(c2cnsn2)=O)C2CC2)C1 Cc1cccc(C(=O)NCC2(CO)CCN(C(C3CC3(C)C)=O)C2)c1C C1(c2n(CCCC)nnn2)(Nc2cnn(C(C)C)c2C)CCOC2(CCOC2)C1 CN1C(=O)C(=O)N(CC(=O)NCCC2(O)CN(C(c3ccnc(O)c3)=O)C2)C1=O C(c1cc(C)cc(C)c1)=CC(=O)NCC1C2N(C(C(C(=C)Cl)(C)C)=O)C(CC2)C1 c1(CN)cn(CC(N2CCCC2C2(NC(N)=O)CC2)=O)nn1.c1cccnc1 C1(CC(=O)NCC(CC=C)NC(c2c(Cl)cnn2C2CC2)=O)CCN(OC)CC1 C1(CC(=O)NCCCCCn2cc(CN(C)C)nn2)CCCC(C#N)C1 c1(OC)cccc(C(C)=CC(=O)NCC(C)N(c2nnc(C(F)(F)F)s2)C)c1 N1(C(c2c(C)occ2)=O)CC2CCN(C(C3(C)CC(C)(C)C3)=O)CC2C1 c1(OC)cccc2c(F)c(COC(=O)C=Cc3cc(Cl)sc3Cl)[nH]c12 c1(CC)cc(C(N2CCCC(CNC(c3cscn3)=O)CC2)=O)cc(Cl)n1 C1(NC(C(F)=CC)=O)CCOC12CCN(C(=O)CSC1CCCCO1)CC2 C1(C(=O)NCCCN(C(C2CCC(CC)CC2)=O)CCO)OCCCC1(C)C c1(CN2CC(C(=O)Nc3cncc(C)n3)OCC2)cn(C)c2ncccc12 CS(=O)CCC(=O)NCC(C)(C)CC1CN(C(=O)Cc2ccccc2CC#N)C1 C(=O)(CC(CCC)C(=O)OCC)NC1(CF)CCN(C(C(C=C=C)C)=O)C1 N1(C(CNS(CC)(=O)=O)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)C2CC12 C1(NC(C2C(C)(C)C2(C)C)=O)CN(C(c2cccc(F)c2N)=O)C2CCCCC12 N1(C(C2N(C)CCC2)=O)CCOCC(F)(CNC(c2ccc(N(C)C)cn2)=O)C1 C1(NC(C2CC(N(C)C)C2)=O)CCC(C)(CNC(=O)C(C2CC2)N(C)C)CC1 CC1(C)CN(C(=O)C(=O)NCCCc2ccc(F)c(F)c2)CCS1 N1(C(C(C2CCCCC2)NC(c2c(OC)n(C)nc2)=O)=O)CC2(CCCN2C)C1 C1(C(=O)NCC(F)(F)C(F)F)(COC)C=CCN1C(=O)C=CC1CCOC1 c1(-n2ccc(C(N3C(C(=O)NCCC)CCC3)=O)n2)ccc(OC)cc1F CC1(F)CC2(CN(C(N3CCCC3n3cc(OC4CC4)nn3)=O)C2)C1 N1(C(C=CC=CC)=O)CCN(CC(=O)NCCc2ncoc2C)CC1 c1(OC(CCC)C)ccc(-c2noc(Cc3ccc(C)cc3)n2)cc1 C12(C(N(C3(C)CN(C(=O)CCC(=O)OC(C)(C)C)C3)C)=O)CCC(CC1)C2(C)C CC(CNCc1csc(C2CC2)c1)CC(C)(C)C N1(C(C(CC#C)C)=O)CC(C)OC2(CCN(C(=O)CCCC(=O)NC)C2)C1 c1(C(N2CCN(C(CC#C)CC(F)F)CC2)=O)c(C)sc2c(Br)cccc12 c1(C(=O)OC)ccc(NC(C2CCN(Cc3cncc(Cl)c3)CC2O)=O)cc1I N1(C(C(C)NC(C)=O)=O)CCC(C)(C)C1CC(=O)N(C)CC1(O)CCCCC1 O=C(C1=COc2ccccc2O1)NC1C=CCN(C(C2C3CCC(F)(F)C23)=O)C1 c1(C(=O)NCC2C(NC(CSc3ccc(C)cc3)=O)C2)cc2oc(C)cc2[nH]1 S(=O)(=O)(CCCN1CCCCC1=O)N(CC(N1CCOCC1)=O)C c1(CN2CCCC(C(=O)NC(c3ccccn3)CCC)C2)cccc(O)c1C N1(C(C2CCC(=O)O2)=O)C2CCC1CN(C(=O)CCOc1cccnc1)C2 C12(C(=O)NC3C(CNC(c4nn(C)c(C(F)(F)F)c4)=O)C3)CCC(CF)(C1)OC2 c1(OC)ccc(Br)c(C(N2CCOCC2CC(N)=O)C(=O)NCCCC2CC2)c1 C(C)(CSC)(C(=O)NCC1(C)CCC(=O)N1)NC(CC(C)N(C)C)=O N1(C(=O)Cc2cocn2)CC2CCN(C(c3ccsn3)=O)C2C1 C=C(C)CC(C(=O)NCC1(NC(=O)C2=C(Cl)CCC2)CCOCC1)OC C(=O)(CC(C(F)(F)F)NC(c1ccc(OC)cc1)=O)NC(CCC=C)C1CC1 c1(C(=O)NCC2CCC(NC(C3C(=C)C3)=O)C2)cccnc1-c1nncn1C N1(C(c2c[nH]c(=N)s2)=O)CCC(NC(=O)CCCc2ncco2)C(CO)CC1 c1(C(N(CC(CNC(c2cc(C)nn2C)=O)(C)C)C)=O)ccc2nccnc2n1 CC(C(=O)NCC1CN(CCN2CCNC2=O)CCCO1)C(F)(F)F C1(CNC(C2C(C=C)C2)=O)CCC(C)(C)CN1C(=O)CSc1ccc(F)cc1F c1(CNC(C(C)SCCCC)=O)cccc(C(N2CC(c3cc(C)no3)C2)=O)n1 Cc1nn(C)c(C(=O)NC23CCN(C(c4c[nH]nc4C4CC4)=O)CC2C3)c1Br N1(Cc2cc([N+](=O)[O-])sn2)CCc2cc(C(F)(F)F)ccc2C1 C1(C(=O)NC(C(=O)N(C)C)CO)CCCCC1NC(C1(Br)CC1)=O Cc1cc(Br)ccc1-n1cc(C(C)NC(=O)CC23CCCC2C3)nn1 C1(CCNC(C(C)N(C(c2cncc(CO)c2)=O)C2CC2)=O)OCCC1(C)C Cc1c(Cl)ccc2c(=NCC3(N(C)C)CCCC3)cc[nH]c12 c1(OC)ccc(CN2CC3CC2CN3C(c2cc(C3(C)CC3)on2)=O)c(F)c1F Cc1cnnc(O)c1C(=O)NCC(=C1CN(C(=O)Cc2ccc(Cl)cc2)C1)F C12(C(N(C)Cc3ccncn3)=O)CCC(CN(C(=O)CN=[N+]=[N-])C1)C2 C(CC(=O)NCC1CC1(F)F)(C(F)F)NC(C1CN(C(C)C)C1)=O c1(NS(CC)(=O)=O)ccc(C(=O)NC(C)C(C2CC2)NC(=O)COCC(F)F)cn1 N1(C(=O)N(c2ccc3c(c2)OCO3)CC(=C)C)C2CCC1CC(N(C)C)C2 Cc1ccc(C(N2CCCC(C)(NC(c3ncoc3C)=O)C2)=O)c(N=[N+]=[N-])c1 N1(C(C(C)(O)C(F)(F)F)=O)CCc2cccc(Br)c2C1.N12C(CC3CC13)C2=O c1(OCC(=C)C)ccc(OCC(=O)N(C(CN(CC)CC)C2CC2)C)cc1 c1(C(N2CCC(NC(COCC)=O)C2)=O)c[nH]n(C2CCCCC2)c1=N N1(C(c2ccc(C)nc2O)=O)CCC(C)N(C(c2cn(C3CCC3)nn2)=O)CC1 N1(C(CC(C)OC)=O)CCC(C)(CNC(c2cccc(C(N)=O)c2)=O)C1 Cc1nc(NC(C2CCCN2Cc2ccc(O)c(O)c2)=O)ccc1O C1(C(N2C(CC(=O)NC(COC)C(=O)OC)CC2)=O)CCOC(C)(C)C1 C1(COC)CN(C(=O)CC2CC2(Cl)Cl)CCN1C(c1ccc(F)c(SC)c1)=O c1(OC(CC)C(N2CCC(C)(NC(=O)C3=C(Cl)CC3)C2)=O)ccc(C)cc1 C1(NC(c2cc(C3CCCC3)[nH]n2)=O)CCC(CNC(C2(Cl)CC2)=O)CC1 C(=O)(C1SCc2cccnc21)NC1CC(NC(c2nnn(CC)c2C)=O)C1 c1(C(=O)NCCC(C)N(C(c2cn(CCCC)nn2)=O)C)coc2c1CSC2 C(CCC(=O)N1CCC(CC(=O)NCCCc2cc[nH]n2)C1)SC C1(CNC(c2scc(C)c2C)=O)CC2(CC2)CN1C(C1OCCN(C)C1=O)=O c1(C(C)C)cc(C(N2CCN(C(=O)Cc3ccc(Cl)s3)CC2C)=O)ccc1O C(=O)(C(C)CC(N)=O)NC(C1CCN(C(C2N(C(=O)OC)CCC2)=O)CC1)(C)C c1(C(N2C3CN(S(c4ccc(CC)s4)(=O)=O)C(C3)C2)=O)cc2cccn2cn1 CCCCCC(F)C(=O)N1CCC(C(C)NC(=O)CN2C(=O)CN(C)C2=O)C1 CCC(F)(F)C(F)F.N1(CCOC)CC(C(c2ccccc2)O)CC1=O C(=O)(CCC(F)(F)F)N(C1CCN(C(C(C)Oc2ccccc2Cl)=O)C1)C C1(C)(CN(C)C(c2ccc(-c3ccccn3)cn2)=O)CCCN1C C=CCC(CC(C)C)C(=O)NCC1CCC(C(=O)NCc2cc(C3CC3)on2)C1 c1(CC2(C(=O)NCCN(C(c3c(C)nn[nH]3)=O)C)CC2)ccc([N+](=O)[O-])cc1 c1(CS(=O)(=O)NC(=O)COC(F)F)cncn1C(C)(C)C C1(C(=O)NCC(=O)NCCN(CC)Cc2ccccc2)CSCC1C.C(=O)(CC)N c1(CN2CC(F)(C(=O)NC(C(CC)C)CO)C2)c(C)[nH]c2ccccc12 c1(C(=O)NCC#CCNC(CN(CCC#C)C)=O)ccnn1CC1CCC1 Cc1cc(F)ccc1C(O)C(=O)N1CC(NC(=O)CCC2CCCCCC2)C1 C1(CC(N2CC(O)(CNC(c3c(C)ccs3)=O)C2)=O)CCCC(C#N)C1 C(=O)(C(C)(C)CC(C)(C)C)NC(CC(CC)C)C(=O)NC1CC(Cl)(Cl)C1 N1(C(Cc2nc(C)sc2)=O)C(CNC(=O)CC2CC(C)OC2C)CC2COCC12 c1(CC)nc(C(=O)NC2CC(NC(c3c(C(C)C)noc3C(C)C)=O)C2)c(C)o1 c1(CC)nc(N2CCOC(C(C)NC(c3oc(C)nc3C)=O)C2)c(CC)c(Cl)n1 c1(C(N(C)CC2OCCN(C(CCCN(C(C)=O)C)=O)C2)=O)cc(C)nc(C)n1 Cn1cc(CC(=O)NC2CCCN(S(=O)(=O)C(F)F)C2)c2ccccc12 C#CCCCCCCC(=O)NC(CCC=C)C(=O)Nc1ccc(OCC)cc1 c1(C(N(C2CN(C(c3cc(OC)c(C)cc3)=O)C2)C)=O)cccc2c1C(=O)NC2 CCCCCS(=O)(=O)CC(=O)NC1CCCC1NC(c1ccc2n[nH]cc2c1)=O C#Cc1ccc(C(N2CCCC2C(C)NC(=O)C=CC)=O)o1 C1(C)(C(=O)NCCC(C)NC(c2ccn(C(C)(C)C)n2)=O)Cc2ccccc2N1 c1(CN(CCCCC)CC(O)CC)ccc(OC)c(F)c1 c1(C(N(C2C(CC)CC(C(=O)O)C2)C2CC2)=O)cnc2onc(C)c2c1 C(=O)(C(C)CC(N)=O)N(CCNC(CCC#CC)=O)Cc1cccnc1 N1(C(C(CC)N(C)C)=O)CCCC(C)(C)C1CNC(c1cncn1C(C)C)=O C1(C(=O)NCCC2(O)CCC2)CCN(C(C2OCC3CCCC23)=O)CCO1 c1(CN2C(C(N(C(c3ccncc3)CC)C)=O)CC2)ccc(F)c(O)c1 N1(C(=O)Cc2ccc(F)c(Cl)c2)CCCN(C(C23CCCC2C3(F)F)=O)CC1 C1(CCNC(=O)COc2ccsc2)CCN(C(=O)Cc2ccccc2Cl)CC1 C1(NC(c2cnc3n2CCS3)=O)COC2(C1)CN(C(=O)CCCCF)C2 N1(C(C=C(CCC)C)=O)CCN(C)CC1CNC(=O)C(CO)OC C1(CNC(C(c2scc(C)n2)(F)F)=O)CC12CCCCC2 C#CC1N(C(=O)C(C)(C)Cc2cn(C(C)(C)C)nn2)CC1(C)C c1(NC(C)=O)ccc(CC(=O)NC2CCN(C(=O)C(CO)N(C)C)C2C)cc1 c1(-c2c(C)onc2)ccc2ccc(C(=O)NCc3c(Cl)cc(Br)cc3Cl)nc2c1 c1(C(=O)NCC2CC(NC(C3C(C(=O)OCC)C3)=O)C2(C)C)c(C)[nH]c(C)c1C C1(C(=O)OC)COC(C)CN1C(CC(=O)OC(C)(C)C)=O.C12(F)CN(C1)C(=O)C2 C(C(O)(CNC(=O)OC(C)(C)C)CO)NC(COC)Cc1ccccc1 N1(C(C(=O)N)C)CCc2c(ncn(C)c2=O)C1.N(CC)CC1CC1 C1(CC(=O)NCCCC(C)NC(=O)CC(C)(C)N(C)C)CCN(C)CC1 c1(CC)cnc(C(=O)NCC2(COC)CCCN2C(=O)C(C)OCOC)nc1 C(c1cccc(Cl)c1Cl)=CC(N1C(CNC(c2cn(C)nc2)=O)CC1)=O C(=O)(CCCCCOCC)NC1CCN(C(C(C)OCC)=O)C1 C1(CC(C)O)CCN(C(c2occc2CNC(=O)CCN(C)CCO)=O)CC1 CC(C)C(F)(F)CC(=O)NCC1CCCCC1NC(c1c[nH]c2ncccc12)=O Cc1nc(F)ccc1C(N1CC2CCC2(C(=O)NCc2c(C#N)cnn2C)C1)=O c1(OC)c(C)cc(C(=O)NC2CC2NC(C2CCC(=O)N2C)=O)cc1Cl c1(OC)cccc(CC(=O)NC2CC(NC(C3CCC(C(N)=O)O3)=O)C(O)C2)c1 C(CN1C(=O)OCc2ccccc21)NC(CNC(CCc1cc(-c2ccc(C)s2)on1)=O)=O c1(C(=O)NCCC2CCN(C(C3(C(C)(C)OC)CC3)=O)C2)cc(C)cc(F)c1N N1(C(c2ccc(C(C)=O)cc2C)=O)CC2(C1)CN(C(C1CCO1)=O)CC2CO c1(C(N2C(c3cn(CCCCCC)nn3)CCCC2)=O)cc2c(s1)CNCC2 N1(C(=O)C(C2CCOCC2)O)CCN(C(c2ccc(O)nc2)=O)CC(O)C1 C1(CN(C(=O)CN2CC=CC2)CC)CCCN1C(c1cncs1)=O C(=O)(C#CC1CCCO1)NCC1(OC)CN(C(CC2(C=C)CCC2)=O)C1 c1(C(N2C(CCC(=O)NCC(CC)C#N)CCC2)=O)ccccc1O CCCCC(O)CC(=O)NC1(C(=O)N(CC(=O)OCCSC)C)CCCC1 C1(C(=O)NCC2N(C(c3cccc(=O)o3)=O)CCN(C)C2)CCc2nnnn2C1 c1(C(=O)NCC(C)N(C(C2CCCC2O)=O)CC)cccc(C(F)F)c1 C(CCC(=O)N1CCC(Oc2ccncc2)C1)C1C(C)C1.C1C(=O)N1 CN1CCCC(O)(CC(=O)NC2CCC(N(C(=O)Cc3cccnc3)C)CC2)C1 CC1CN(N2CCCC(OCCO)C2)Cc2n[nH]cc21 N12CC=C(CCNC3(CCC3)C1=O)CC2.c1(CC(=O)OCC)cc(C2CC2)no1 CCC(O)C(C)C(=O)NC1CCC(CNC(=O)CCC2CCC2)C1 c1(CNC(C)=O)cccc(S(=O)(=O)N2CC3CC(F)CC3C2)c1 CN1CCCC(F)(C(=O)NC2CC(NC(=O)C(c3cccc(F)c3)O)C2)C1 C(=O)(C(CCC(C)C)NC(C1CC(C)CC(C)(C)C1)=O)NCC(CC=C)(C)C CN1CCC(O)C(NC(=O)CC2CCN2C(=O)CN2CC=CC2)C1 c1(OC)cc(O)c(C(=O)NC23COC(C2)C(NC(=O)CC(C)CF)C3)cc1OC C1(C)(C(=O)OCC2CC(OC)C2)CCCCC1(F)F C1(C(=O)Nc2c(SC)cc(Cl)cc2)CC1C1(C)CCCN(Cc2ccc(Br)cc2)C1 C1(C(=O)NCCOC2CCN(C(C(C)SC)=O)C2)CSC(c2ccccc2O)=N1 c1(N2CCCC(NC(c3cnn(CCF)c3)=O)(CO)C2)c(Cl)cccc1[N+](=O)[O-] C1(N(C)C(C2CC(c3cncn3C)=NO2)=O)CS(=O)(=O)C12CCNCC2 n1(CC(C)NC(C2CCC(CSc3nonc3N)CC2)=O)ncc2ccccc12 C(=O)(C(C)(COC)CC)NC1C(CNC(C(c2ccc(OC)cc2)=O)=O)C1 C(=O)(CCC(=O)N1CCCCC1C(N1CC2CC2C1)=O)OCC C=C(C)CC(C(=O)N1CC2CC2(CNC(C2CC23CCCC3)=O)C1)NC(C)=O C1(O)(CCNC(c2c(C)nc(N(C)C)s2)=O)CCN(C(C2CSCCS2)=O)CC1 C1(C)(C(=O)NC(CNC(c2ccc(OC(C)C)nc2)=O)CO)CCC(=O)N(C)C1 Cc1cc(C(=O)NC2CC(C(=O)NCc3cccnc3)CC2O)nc(O)c1 C1(CNC(Cc2cccc(C)c2)=O)CC2CC1CN2C(c1cc(C#N)c[nH]1)=O C(CC(=O)NCc1cccc(NC(=O)CC2CC=CCC2)c1)(C(F)(F)F)OC N1(C(CC(C)(C)O)=O)CCOCC(F)(CNC(=O)CC2(CO)CCCC2)C1 N1(C(C(CSC)(C)C)=O)CCC(NC(C2CCN(c3ccncc3)C2)=O)C(O)C1 C1(CC(=O)NC2CCN(C(CCc3c(C)c[nH]c3C)=O)C2)CCC(C)(C)CC1 C(C(=O)C(C)N1CCC(C(F)F)C1)NC(=O)OC c1(NC(C2N(Cc3cc(C)cc(F)c3)CC(O)C2)=O)ccc(Br)c(Cl)c1C Cc1ccc(NS(C)(=O)=O)c(C(N2CC(NC(=O)CC3CSC3)CC(C)C2)=O)c1 N1(C(C(C)S(N)(=O)=O)=O)CC(CO)C2(C1)CN(C(=O)CN(S(C)(=O)=O)C)C2 c1(C(=O)NCC(C2CC2)NC(C2CC(F)(F)C2)=O)ccc2nc(C3CC3)oc2c1 c1(OCC(N2CCC(NC(C3C(C=C)CC3)=O)CC2)=O)cc(F)cc(F)c1 C(C(O)C(F)(F)C(F)(F)F)NC(=O)CN(CC(=O)OC)C C(CC1=CCN(C(=O)CC2(O)CCCOC2)CC1)NC(c1cc(Cl)nnc1Cl)=O C1(CNC(=O)Cc2c(F)cccc2F)CCC2(CCN(C(=O)CO)CC2)O1 CN=c1ccc(C(N2CCCC(CCNC(=O)CC3CC(C)=NO3)C2)=O)c[nH]1 N1(C(C)=O)CS(=O)(=O)CC1C(N1CCN(C(c2cnn(C)c2Cl)=O)CC1C)=O C=C(C)CCC(c1nnnn1CC)NC1(c2nc(-c3ccccc3)no2)CC1 c1(NC(C(=O)NCC(c2ccc(Cl)cc2)OCC)=O)ccc2ccsc2c1 C1(CNC(c2c[nH]nc2C(F)(F)F)=O)CCN(C(C2(c3cccs3)CC2)=O)C1 C1(F)(C(=O)NCCCN(C(=O)Cc2ccccc2C(C)C)CC)CC=CCC1 C1(NC(CC2(NC(C(C)NC(=O)C3CC3)=O)CC2)=O)C(C)CCC1C C1(C(=O)NC2CCC(F)CC2)(CC)CCN(C(c2ccc(Cl)o2)=O)C1 C#Cc1cccc(C(=O)NCCC2CCCN(C(=O)CC(CC)SC)C2)c1F c1(C(N(CC(C)NC(C2(N(C)CC)CCCC2)=O)CC)=O)cc(C)n(C)n1 C(C(=O)NCCN1CCOCC1)(C1=NOC2(COC2)C1)N1CC(CC)SCC1 C1(NC(=O)CC23CCCC2C3)CCCCN(C(=O)Cn2ccc(O)nc2=O)C1 S(=O)(=O)(c1ccc(=NCc2cccnc2F)[nH]c1)NCC1C(C)(C)C1 C1(NC(c2cc(C)c(C)s2)=O)CCCCCN(C(C2CCCCC(=O)N2)=O)C1 C(=O)(CCC(C)(C)C(=O)OC(C)(C)C)N1C(CNC(C2CC(SC)C2)=O)CCC1 CON(CCC(=O)NCc1nocc1Br)C(=O)c1c[nH]nc1Cl N1(C(C2N(C)CCOC2)=O)C2CCC1CN(C(C1(N(C)C)CCC1)=O)C2.C(C)(C)N C12(C(NOCC(=O)N(CCC(C)C)C)=O)CCC(C1)OC2C C(CC(F)F)(C(=O)N1CCC1(C)C(C)C)NC(C(CCOC)C)=O C1(C(N2CCC(CC)C2)=O)C2CN(C(c3cn(C)nc3C(F)F)=O)CC12 c1(C(N(CCNC(C2CC(CCC)OCC2)=O)CCC)=O)cc(S(N)(=O)=O)co1 c1(C(=O)NCC2CCCC(NC(C3(C)CC=CC3)=O)C2)cc2ccccc2o1 N1(C(CC(C)CC(F)(F)F)=O)CCC(O)(C2(NC(c3cnn[nH]3)=O)CC2)CC1 C1(CC=C)(NC(=O)C=Cc2ccncn2)CCCN(C(C2CCC(=O)NC2)=O)C1 C(=O)(CC(C)(C)CCOC)NC(C(C)NC(C1(C=C)CC1)=O)(C)C N12CCCC(C)(C1)C(=O)N(CCOC)CC2=O.C1(CN(C)C)CC(F)(F)C1 C1(CNC(C(N2CCCC(C)(C(F)(F)F)C2)=O)=O)CCCC2CCCN12 CCCCCCC(=O)N(C1CCCC1)CCNC(c1cccc(OCF)c1)=O C1(C)(CNC(C=C(C)C)=O)CN(C(=O)CC2CC3(CCCC3)CO2)C(C)(C)C1 c1(NC(CC2(C)CN(C(=O)NCCCl)C2)=O)ccc(Br)cc1[N+](=O)[O-] C=CCCCC(C(=O)NCC(O)C(=O)NCCC=C)NC(=O)C(CC)OC CCC1=NOC(CC(=O)NCCCC(=O)NCCc2ccnc(C)c2)C1 Cc1cc(O)ccc1C(=O)NC1CC(CCNC(=O)Cn2cc(C(F)F)cn2)C1 C1(O)(CNC(c2cc(CC)on2)=O)CCN(C(C2CC(=O)CO2)=O)C1 C(CC(C)C)(C=O)OC.C1(C(N)=O)COC(CN2CCC2C(=O)OC)C1 C(=O)(CCS(N)(=O)=O)NCC(=O)NC(C)(C)C(N1C(CO)CCC1CO)=O C1(NC(c2c(OC)ccc(F)c2N)=O)CN(C(CNC(CC)=O)=O)CC(F)(F)C1 C(=O)(C1CCc2ccccc21)N1CC(CCCC)N(C(c2cc(C)on2)=O)CC1 C1(NC(C(C)OCC2CCCO2)=O)CN(Cc2nnc(O)s2)CCC1C C1(C)(CNC(C23CC(C)C2C3)=O)CCCN1C(c1cc(C(F)F)[nH]n1)=O C1(C(=O)NC2C(NC(c3c(CC)nn(C)c3)=O)COC2)CCC2(CCCCC2)C1 Cc1cc(C(=O)NCC2(C(N)=O)CN(C(c3cnn(C)c3C)=O)C2)sc1C N1(C(c2cc(CC)n(C)n2)=O)CCC(Nc2ncccn2)C(O)C1 CCC(C)C(C)C(=O)NC1CCCCC1NC(=O)Cc1sc(C)cc1C c1(SC)nc(NC(C2CC(O)CN2C(=O)Cc2ccc(Br)cc2Br)=O)ncc1F C(=O)(C(C)CCOC)N(CCCNC(c1cccc(=O)o1)=O)CC c12ccc(cc1)OCC1(CN(C)C1)OC(=O)CO2.c1(N(C)C)ncccc1F.C(O)N C=CCC(CNC(C1OCCC1C)=O)C(=O)Nc1c(CC)noc1C C1(NC(c2cc(CCC)on2)=O)CC2CC1CN(C(C1(CC(C)C)CC1)=O)C2 c1(C(=O)NCCCN(C(C)C)C(c2ccncc2Br)=O)cc(O)cc(F)c1 CC1CN(C(=O)CNC(=O)CC2CC3CCC2O3)CCC1(F)F c1(C(=O)NC2CCN(C(CCCCOC)=O)CC2CO)nc(Cl)cc(N)c1Cl c1(C(N2C(CNC(c3cc(C)no3)=O)C(C)CC2)=O)cc2ccccc2o1 n1(CCCCCC)c(-c2nc(-c3ccnn3CC)cs2)nc2ccc(F)cc2c1=O c1(C(N2CCCC(CC(=O)OC)C2)C(=O)NCCC#N)nc2c(s1)CCCCC2 c1(C(=O)NC2C(CNC(CNC(=O)OC)=O)CCC2)cccc2c1C(F)(F)CC2 N1(C(CCCC#N)=O)CCC(NC(c2cc(Cl)ccc2C(F)F)=O)C(F)C1 C1(C(=O)NC2CN(C(C(CC)C#N)=O)CC2CO)CN2CCC1CC2 C(=O)(C(F)CC(C)C)N1CC(NC(c2cn(CCOC)nc2C)=O)C(OC)C1 C1(NC(CC2C=NN(C)C2=O)=O)CN(C(c2csc3nccn23)=O)CC12CC2 c1(C(N2CCC(C)(NC(c3cc(C)c(C)nc3)=O)C2)=O)nccc2occc12 Cc1cc(CNC(C2CNC(C)(C)C2)=O)cc(C)c1Cl C=CC(C)(O)C(=O)NC(C)(CNC(c1cnnn1C1CC1)=O)C1CCC1 N1(C(C(CC#C)(C)NC(c2ccc[n+]([O-])c2)=O)=O)CC(O)CC(C)(C)C1 c1(C(N(C(CNC(c2nncc(OC)c2)=O)C2CC2)C)=O)ncnc2ccsc12 C1(CC(=O)NCCC(C)NC(=O)CCCc2cccc(Cl)n2)CC2(CCC2)CO1 N1(C(COCC(=C)C)=O)CC2(C1)CN(C(=O)Cc1cc(C)cc(F)c1)CC2CO N1(C(c2ccc(C)cc2)=O)C2CCC(C2)C1C(=O)NOCC(O)CO O=C1CC2(C(N3CCC(C(=O)O)CC3)=O)CNCC2N1 c1(C(C)=O)ccc(=NCC2CCCCC2NC(C2CC3CCC(C2)S3)=O)[nH]c1C C1(NC(C(CSC)OC)=O)CC(O)CN(C(=O)CC2(C)CC2)C1 N1(S(c2cccc(OC)c2Cl)(=O)=O)CCc2nc(C)nc(O)c2C1 c1(C(N2CCCC2(C)CCC(=O)O)C)cc(I)c(F)cc1F CCCC(CCCNC(=O)CCCOC)NC(=O)CC1CC(C2CC2)C1 C(C)(C(=O)NOCC(F)(F)F)N(CCC)C(c1cc(C(C)=O)[nH]n1)=O C12(CNC(C(n3cnc(C#N)n3)CC)=O)CC(NC(c3ccsc3C)=O)(CO1)C2 N1(C(C=CCN(C)CC)=O)CCCC(CC)C1CNC(=O)CC=CC(C)(C)C CN1CC(=O)N(CC(=O)NCC2CCCC(NC(=O)Cn3nccn3)C2)C1=O Cc1ccc(CC2CCN(C(CSN(C(=O)COCCCF)C)=O)C2)cc1C C1(NC(C(CC)N(C)C)=O)COCCC1NC(C1CCCNC1=O)=O N1(C(CCCCSC)=O)CCC2(CCCN(C(=O)Cc3cnc[nH]3)C2)CC1 c1(C(=O)NCC(c2cc(C)oc2C)(C)O)cc([N+](=O)[O-])ccc1O CC(C(=O)NCCOCCOCCCNC(C1(C)CCC1)=O)C1CCC1 CCC(C)(F)C(=O)NCc1cn(C2CCN(C(=O)C(F)(F)CC)C2)nn1 N1(C(CCN(C(=O)C=Cc2ccco2)CC2CC2)=O)CCOC2(CC2)C1 C(CCCCC(=O)Nc1cccc(CNC(=O)CCC2CCCC(=O)N2)c1)OC c1(SC)ccc(C(=O)NC2COCC2NC(C2CCOC2C(C)C)=O)s1 c1(CC)nc(C(=O)N(CC(=O)NC(C2CCN(C)C2)C)C(C)C)co1 N1(C(CCNC(=O)OCC)=O)CC=C(CC(=O)N2CCC2C(=O)OC)CC1 c1(N(C(C2CCN(C(=O)C(CN(C)C)N(C)C)C2C)=O)CC)ccc(C)nc1 C1(C(CC)NC(C2NCCC2c2ccccc2)=O)CCC(F)(F)CC1 N1(C(C(CC=C)OC)=O)CCC2(CC2)CC1C(=O)NC(CO)C1CC1 c1(NC(Cn2cc(-c3cnc(C)o3)nn2)=O)ccc(Cl)c(I)c1 CCC(C)(CNC(=O)C(CNC(=O)CCC1CC1C)OC)C(N)=O C(=O)(CC1C(=O)Nc2ccc(F)cc21)N1CC(CCNC(C(C(CC)C)O)=O)C1 Cc1nn(C)c(Cl)c1C(N1CC2(CNC(=O)CC3C=NN(C)C3=O)CCC1C2)=O CN1CCC(C(=O)NCC(C(C)(C)C)NC(=O)OC(C)(C)C)C(C)(C)C1 N1(C(CCCOC(C(C)C)=O)=O)CCC(C(CO)NC(=O)CC2CC2CF)CC1 O=C1CCN(C(C2CCN(Cc3ccc(F)cn3)C2)=O)CCN1 c1(C(=O)NC2C(NC(C(C)OCC)=O)CCC2)c(N)cc(Cl)nc1Cl c1(NC(=O)NC2CCCN(C(C)(C)C)C2=O)ccc(S(N)(=O)=O)cn1 C1(NC(Cc2nnc(C3(OC)CCOC3)o2)=O)Cc2ccccc2C1(C)C C1(C(N2C(CNC(C3(c4onc(C)n4)CC3)=O)CCC2)=O)C2CC3C(C2=O)C13.COC N1(C(CCCOCC=C)=O)CC2CC(C1)N(C(=O)C=CSc1ccccc1)C2 CC1(CNC(C2CCNC(=O)C2)=O)CCCN1C(=O)CC1C=CS(=O)(=O)C1 C(=O)(CC(C(F)(F)F)NC(c1cccc(CC#N)c1)=O)Nc1ccc(CC)cc1 N1(Cc2c(C)csc2)CCOC(c2ccnc(N3CCC3)n2)C1 N1(C(CCCC#C)C(=O)Nc2c(C)cc(C)cc2C)CCc2c(F)cccc21 CC(C)C(C(=O)NCC(C)N(C(=O)C(C)NC=O)C)C1CCC1 C1(O)(CN(C)C(C2CCCCN2S(C)(=O)=O)=O)CCN(C(=O)C=CC2CCC2)C1 C1(C(N2CCCC(NC(C(C(C)C)O)=O)C2C)=O)CC2COCC(C1)C2 C1(C(N(C(C)=O)Cc2nc(C)cs2)=O)N(C(c2scc(C)c2C)=O)CCC1(C)C C1(CC)(NC(=O)C=CCNC(=O)CCn2ccnc2C)CCCCCC1 n1(CC(=O)NCC(C)NC(=O)Cn2cc(C3CC3)nn2)cc(Cl)c(O)nc1=O c1(OC)ccccc1C(O)C(=O)N(CC(O)CN(C)C(c1ccc(Cl)o1)=O)C c1(OC(C)C)nc(C(c2cncc(N(C)C)c2)C2CC2)n(-c2ccc(F)nc2)n1 c1(C(=O)OCC(=O)C2(c3ccno3)CC2)ccccc1Br c1(NCC2C(C)C2(F)F)ncccc1S(=O)(=O)NC1CCn2nccc2C1 CN1CCN2CCN(C(=O)N(CC(C)(C)C)C)CC2C1=O n12ccc(cc1=O)CS2.C1(CC(=O)N(C2(C(C3CC3)OC)CC2)C)CCC(=O)O1 N1(C(=O)Cn2ncc(O)nc2=O)CCCCC(NC(c2ccc[n+]([O-])c2)=O)C1 Cc1cc(C(=O)NC2CC3CN(C(=O)CC4CN(C)C4)CC3C2)ccc1[N+](=O)[O-] Cc1cnc2n1CCC(C(N1CCC(O)(CNC(=O)Cc3nc[nH]n3)CC1)=O)C2 N1(C(CC)=O)CC2CC1C2C(=O)NCC(C)(O)CCO Cc1ccc(CN2CCC(O)(C(N3CCC(c4nc(C)no4)C3)=O)CC2)c(Cl)c1 CCC(CC(F)(F)F)C(=O)NC(C)(CNC(=O)Cc1cccnc1C)CC1CC1 c1(SCC(=O)NC2CN(C(C(C)=C(C)C)=O)CC2C(F)F)ccc(C)cc1C c1(C(N2CC(C)C(CNC(=O)C(C)CC(N)=O)C2)=O)ccc(F)c2ccncc12 C(C(C)(C)C(=O)NC(C)CCCCNC(=O)CC1CCCC1)SC c1(CC(=O)NC(C)CCNC(c2cc(C(F)F)[nH]n2)=O)nnc(S)n1C C(=O)(CC(CC)C(C)(C)C)NCC(CCC)NC(C=CCCC)=O c1(C(N2CC(CC(C)NC(C(CC(C)C)OC)=O)C2)=O)ccc2oc(=O)oc2c1 C#CCC(C)(C)C(=O)NC1CC(NC(c2c[nH]nc2C(F)(F)F)=O)C(O)C1 C1(CNC(C2(O)CCSC2)N(C)C)C2CN(C(=O)CC3CSC3)CC12 C1(C2CC2)(CNC(=O)C=C2CCCCC2)CCN(C(=O)CC2CC2)C1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1NC1CC1)N1C(C)C(O)CC1 CP(C)(=O)C1CCC(=CCOC(c2cccc(CN3CCCC3)c2)=O)C1 c1(OC)nc(NC2CC2C(=O)Nc2c(Br)cnn2C)nc2[nH]cnc12 N1(C(Cn2c(C)ccn2)=O)CC(CCNC(=O)Cc2cc[nH]c2)OC(C)C1 c1(-n2c(C(=O)NC3CC(c4ccccc4F)(O)C3)ccn2)cccc(F)c1 C(=O)(NN1CCN(C)CC1)n1cc(C2CCCN(C(C)=O)C2)nn1 C=C1CC2(C1)CC(C(=O)NCC(CC(C)C)NC(=O)C=Cc1ccccn1)C2 C1(C(N2CCOCC(NC(c3nc(CCC)oc3)=O)C2)=O)CN2CCCC2CO1 C1(C(=O)Nc2cnn(C(C)C)c2)(NC(CCC)=O)CCSC1 C(=O)(CC1=CCOCC1)NC(C12CCCC1C2)C(=O)NC1CC(C)C1 C1(CC)CCCCC1OCCCC(=O)N(CC(=O)NC)C(C(=O)NC(C)C)CC Nc1cccc(C(F)F)c1C(=O)NCC1(F)CCN(C(=O)C(O)C(F)F)CC1 c1(C(N2CCOC(CNC(C34COC(C3)C4)=O)C2)=O)ccc2ncnn2c1 Cc1ccc(C(F)(F)C(=O)NC(C)C(C)NC(=O)COCCc2cccs2)nc1 c1(NC(N2CC3C(C)C3C2)=O)cc([N+](=O)[O-])cc(Br)c1F Cc1ccnc(N(C2CNCC2C#N)C(c2cnc(C3CCCC3)nc2)=O)n1 c1(C(N2CCC(N(C(CCC=C)=O)CC)C2)=O)[nH]c(C)c(C(C)=O)c1CCC c1(C(=O)NC2CCCN(C(C3CC=C(C)CC3)=O)C2C)cc2[nH]nc(C)c2cn1 C=CCC(C(=O)N(CC)CC1CCN(C(=O)Cc2csnc2C)C1)OC CC1CC(NC(=O)CSc2ccc(F)cc2)CN1C(=O)C(C)CSc1nccs1 Cc1ccc(C(N2CC(NC(c3occ4c3CCC4)=O)C(C)C2)=O)c(F)c1F Cc1cccc(C(=O)NC2CCC(C)(CNC(=O)CCCc3ccsc3)C2)c1 n1(CCOCCNC(c2ccsn2)=O)cc(CCN(C2CCOC2)C)nn1 C1(C(=O)NC2C(NC(c3ccco3)=O)CCC2)CCC(F)(F)C1 C(=O)(CS(=O)(=O)C(C)C)N1C(C(=O)NC2CC(CC3CCC3)C2)CC(OC)C1 CC#CCCC(=O)NC1CN(C(c2nc(Cl)oc2C)=O)CC1C CCCCC(CC)C(=O)N1CC2CCC1(CNC(c1ccnnc1O)=O)CC2 CCCCCC(C)CC(=O)NC1CC(NC(c2c(C)nc(=N)[nH]c2C)=O)C1 C1(CC(=O)NC2CCCC(N(C(=O)COCCF)C)C2)(COC)CCOCC1 c1(C(=O)NC2(CN(C)C(C3CC(=O)N(O)C3)=O)CC2)ccc(C2(C)CC2)cc1 C1(C(=O)NCC(CN(C(c2cnc(C)o2)=O)C)C)C2CCCCC12 c1(C2CCCC(=O)N2)ccc(Cl)cc1.C1(CC)(NC)COC1 C1(C(N2C3C(CNC(c4nc(Cl)cs4)=O)C(C3)C2)=O)CCC2C1C2(F)F N1(C(c2ccc(CC)o2)=O)CCN(C(C2CCC23CCC3)=O)C(CCOC)C1 C12(C)CCN(CC1)C2=O.c1(C(=O)NC)cccc(-c2ccc(OC(C)C)nc2)c1 c1(C(=O)NC(CC(C)NC(C(CC)(F)F)=O)C)cc2sc(Cl)cc2[nH]1 C(c1cccc(O)c1)=CC(=O)NCC1CCCN(C(C2(C=C)CC2)=O)C1 CCC(C(=O)NC1(C(=O)NCC2(C3(O)CCC3)CC2)CC1)C(=O)c1ccc(C)cc1 Cc1ccc(F)c(C(F)(F)C(N2CCCCC(NC(C3CC34CCC4)=O)C2)=O)c1 C(C(C)(C(=O)N(CCO)CCO)NC(=O)Cn1cc(Cl)cn1)SC c1(NC(c2cc(F)ccc2-c2cccnc2)=O)cnn2c1OCCC2 N1(C(c2ncn(CC)n2)=O)CCC(C(F)(F)F)C(NC(=O)C2=NOCC2)C1 N12CC(C1)CNC(=O)C1(CC1)C2=O.C1(CC=C(C)C)(OC(C)=O)CC1 C1(CCNC(c2c(CNC(c3c(C)non3)=O)ocn2)=O)CCN(C)C1=O c1(C(N2CCC(N(C(C(CCC)C#N)=O)C)CC2)=O)ccc2c(c1)CC(C)(C)O2 CCC(CO)(C(=O)NCC1(C)CN(C(=O)CC2CCC2C)CCO1)OC c1(C(=O)NC(C)(CNC(=O)CCS(C)(=O)=O)C2CC2)nccc2n[nH]cc12 CCCC(=O)NCC(=O)NCCCNC(=O)NCC(C)(C)C1CCCO1 C(C(CC(C)C)C(=O)NC(C1CCCCC1)C)NC(c1ccnc(C)c1C)=O c1(C(N2C(CN(C(=O)CCS(C)=O)C)CCC2)=O)cc(F)cc2ccoc12 C1(CCC)CN(C(c2cc[nH]n2)=O)CCN1C(c1ccnc(O)c1Br)=O c1(OCC#C)ncccc1C(=O)NC1CN(C(C2CSCN2C)=O)CC1C CC(C)CCC(=O)NCC1(C)CCC(NC(c2coc(Cc3ccccc3)n2)=O)C1 C(Cc1ccccc1)(CCNC(c1ccn(C)n1)=O)NC(C(C)=C1CC1)=O C(=O)(C(CC)(CC)OC)NC(CNC(Cc1cn(CC)nc1)=O)CCOC C(=O)(CC(F)(F)C(F)F)N1CCC(CNC(c2ccn(C)c2)=O)C1 c1(C(N(CCOCCNC(CC=CCC)=O)C)=O)cccc(N)c1O C1(NC(C2(C(=O)NOCCC3CC3)CCC2)=O)CC2(CO)COC1C2.NC=O N1(C(c2cc(C)cc(O)n2)=O)CCC2CN(C(C34CC=CCN3CCC4)=O)CC12 c1(N2CCC(CNC(=O)C(c3ccccc3)O)C2)ccccc1[N+](=O)[O-] c1(C(=O)OC)n[nH]c2cc(OC(=O)CCc3cc(F)ccc3Br)ccc12 c1(OC)ccc(NC(=O)Nc2ccc(N3CCCS3(=O)=O)cc2C(F)(F)F)cc1 C(=O)(C(C)CC1CCCN1Cc1ccccc1)NC(C)C.C12(CC1)C(=O)OC2 O=S(=O)(c1c(Cl)nc2cc(Cl)ccn12)NC1CC(S(=O)(=O)C(F)(F)F)C1 c1(C(=O)NC2CN(C(c3ccc(OC)c(Cl)c3)=O)C2)sc2ccccc2c1Cl N1(C(C2C(=C)C2)=O)CCC(c2cc(CNC(c3ccc(C)o3)=O)on2)CC1 CC1CN(C(C2CC3(C2)CC3(F)F)=O)CCC1NC(c1cc(CN(C)C)c[nH]1)=O c1(CC2(C(N(C3CCN(C(COCC(C)C)=O)C3)C)=O)CC2)cccc(F)c1 Cn1cc2c(n1)CCCC2C(=O)N1CCC(NC(c2ccc(Br)o2)=O)CC1 CC(C)C(CCNC(=O)CCc1cccc(O)c1)NC(=O)CCCc1nc[nH]n1 N1(C(C(C=CCCC)O)=O)CCCCC2(CCN(C(C3(F)CC3)=O)C2)C1 C1(CNC(=O)CC(=O)NC2CC2)CC2(CCN(C(=O)Cc3ccsn3)C2)CO1 C(=O)(CCCC(C)c1cccc(OC)c1)N(CCCNC(=O)C(C)C1CC1)CC C1(C(N2CCCC(CNC(C3C(C(C)C)CCC3)=O)C2)=O)CCc2n[nH]cc2C1 C(=O)(CCC(CF)CF)N(CCCCNC(C(C)NC1(CO)CCCC1)=O)C c1(SC)ccccc1CC(N1CC(O)(C(C)NC(c2ocnc2C)=O)C1)=O C#CCC(C(=O)NCC1C2CN(C(c3cnn(C4CC4)c3Cl)=O)CC12)C1CC1 C1(C(N(C(C)CNC(=O)CSc2nnnn2C2CC2)C)=O)C2CCCCC12 c1(CC(=O)NCC2(c3ccccc3)CC2)ccc(-n2cc(C3CC3)nn2)cc1 C1(NC(=O)C2=CCCC2)CC(F)(F)CC1NC(c1cnco1)=O N1(C(C(c2ccc(C)cc2)=O)=O)CCCC(C)(CNC(=O)C(C)c2ccco2)C1 CC1CCC(C)N1C(c1nc(C(=O)NCc2cccc(I)c2)cs1)=O c1(C(N(C2CCCN(C(c3cccn(C)c3=O)=O)CC2)C)=O)cc(O)cc(=O)o1 C1(CNC(C)=O)CCN(C(C23CCC(C2)OC3C)=O)CC1C CCCC(C(=O)NC1COCC1NC(=O)C(c1ccccc1F)F)OC N1(C(C(=O)N(C2CC(CN)C(O)C2)C2CC2)=O)CCCC2NC(=O)CC12 N1(C(C)OC2CCOC2)CCC2(CCCC2N=c2[nH]nc(C(C)(C)CCl)o2)CC1 N1(C(COCCN(C)C)=O)CCC2C(C(=O)NCC3C=CCCC3)C2C1 O=C(C1CCCn2nccc21)NCC1C2CN(CC(=O)NCCO)CC12 N1(CCCC)CCCCC1C(=O)NCCC1CN(C(=O)CC2CC(=O)C2)CCO1 C12(C(=O)NC34C(CN(C(c5cccc(CCC)c5)=O)C3)C4)CCCC(CO1)C2 N1(C(=O)NCc2cc3n(n2)CCO3)CC2CCC2(CCF)C1 N1(C(COCC(C)C)=O)Cc2ccccc2C(NC(C23CC(C#N)(C2)C3)=O)C1 c1(C(CNC(C(CCC)OC)=O)NC(=O)CC(C)(C)O)ccc(F)cc1F N1(C(c2nc(C(=O)OCC)sc2)=O)CCCC2(CCO2)C1 CC(C)(Cc1cn(CC2CCCN2C(c2cn(CCO)nn2)=O)nn1)CO c1(C(=O)NC(C(C)NC(CN2CCC(C)CC2)=O)C)cc(S(N)(=O)=O)cs1 Cc1nc(S(=O)(=O)Oc2ccccc2COc2ccc([N+](=O)[O-])cc2I)cn1C N1(C(CC2C(C)=NNC2=O)=O)CC(C(=O)NC2(CC(C)C)CC2)C(C)(C)C1 C=C(C)C1CN(C(c2csc(-c3ccoc3)n2)C(=O)NCC2CC2)CCO1 C(=O)(CC(O)C(C)C)NCC1C(C(=O)Nc2c(C)ccnc2)OCC1 CC(=O)CCCCC(=O)N1CCCCC2CC12 C1(NC(=O)NC(C(C)OC)C)CCC(N2C(=O)CCC2=O)CC1 c1(OC)c(F)ccc(C(N2CC3CC2CN3C(=O)CC2CCC(=O)N2)=O)c1F N1(C(c2cc(Cl)c(Br)cn2)C(=O)NCCN2CCOCC2)CCc2c(Cl)cccc21 N1(C(C(C)C)=O)CCc2c(C(N3CCC(C(C)N(C)C)CC3)=O)csc2C1 C(=O)(CP(C)(C)=O)N1CCC(C2N(C(C3(c4ccn(C)n4)CC3)=O)CCC2)C1 c1(C(=O)NCCCN(C)C(C2(CF)CC2)=O)ccc(O)nc1Cl N1(C(CCOCC(N2CC(C(=O)OC)(COC)C2)=O)=O)CCOC(CC(C)C)C1 N1(C(C#CC2(C)CC2)=O)CC(NC(c2c[nH]cc2Br)=O)C2CCCCC12 c1(NC(C(C)N(C(C(CC)n2ccnc2)=O)C)=O)c(C)n[nH]c1C C1(C)(CNC(C(C)NC(CC)=O)=O)CCCN1C(C1CCC(C(N)=O)CC1)=O Cc1c(F)ccc(Cl)c1C(=O)NCC1(CNC(C2CCC(F)C2)=O)CCOCC1 c1(CC)cccc(F)c1C(=O)OCC(=O)CCCOC C1(CCC)COCCN1C(=O)C(C1CCC1)NC(=O)C(C)=C1CC1 C(=O)(C1CC(C)c2c(C)cccc21)N1CC(O)(CNC(c2ccc(CC)o2)=O)C1 N1(C(C(CC#C)(C)C)=O)CC23CCCC2(C1)CN(C(=O)CC1CCN(C)C1=O)C3 C1(C(=O)NC(c2nn(C)cc2O)C)CCCN(C(c2cccs2)=O)C1 c1(C2N(C(CC3(C(=O)OC)CC3)=O)CCC2)c(C)noc1C C1(CC(=O)N(C(C)C)CCNC(=O)CCNC(c2ccoc2)=O)NC(=O)NC1=O N1(C(C(C)NC(C(C)OCCC(C)C)=O)=O)CC(C2CCC2)C1 c1(OC)cc(CNCc2ccc(S(N)(=O)=O)cc2Cl)c2c(c1)CC(C)O2 c1(C(=O)NC(C2CCCN(C(C3CCCSS3)=O)C2)C)cccc2ccncc12 C1(SC)CCN(C(=NCCOC(F)F)NCc2ccc(F)cc2OC(F)F)CC1 c1(CC(C(=O)OC)NCCc2ncc[nH]2)ccc(C(F)(F)F)cc1 c1(C(N2CC(NC(c3c(C)nccn3)=O)C(C)C2)=O)cccc(Cl)c1O c1(C(=O)NC2CCC(CCNC(C(C)=CC)=O)C2)cnn2c(OC)cccc12 c1(C(N2CCC(C)C2NC(c2ccccc2)=O)=O)n[nH]c2c1CCOC2 C1(C)(CNCc2cccc(OCCOC)c2)CCC(=O)NC1 C1(NC(C(=O)N(CC(C)(C)C#N)CC)=O)NCCC1C1CC1 C1(C)(CC)CC(NC(=O)CC(C)(C)CN(C)C)CN1C(=O)C(c1ccc(Cl)s1)=O N1(C(CC(C)SC)=O)CCC(C(C)NC(c2cnn(C)c2C(C)C)=O)CC1 C1(NC(c2c(C)nco2)=O)CC2(C1)CC2C(N1CCCC(CC(C)C)C1)=O C1(C2CN(C(=O)CC3OCCO3)C2)(NC(C2C(c3ccc(CC)cc3)C2)=O)CC1 C1(NC(=O)Cc2cc[nH]c2)CCCCCCC1NC(=O)C(O)Cc1ccccn1 c1(CCC)ncoc1C(=O)N(CC(=O)NCC1(CO)CCCC1)CC(C)C C(=O)(C(CC(N)=O)NC(C12CCCC1C2)=O)NCCCNC(C(C)C)=O c1(C(=O)NCC(C)N(C(=O)Cc2cnns2)C)cc(Cl)c(O)c(Cl)c1 N1(C(CS(CC)(=O)=O)=O)CC2CCC(C1)N2C(c1cccc2[nH]ccc12)=O C#CCCCC(C)C(=O)NCCCCCCNC(c1ccc(C#C)nc1)=O c1(OC)cc(C(=O)NC2CCCC(NC(c3ncn(C)n3)=O)C2)ccc1Br c1(C(C(=O)OCC)(F)F)ccc(NC2(CC(N)=O)CC2)c([N+](=O)[O-])c1 N1(C(c2c(C)nns2)=O)CCCC2CN(CCCOc3ccccc3)CC12 Cc1ncc(C(N2CC(NC(C3OCC3(C)C)=O)C(C(F)F)C2)=O)cn1 C1(C(=O)NCc2nc(C(N3CC(c4cc(O)no4)C3)=O)co2)OCC2CCCC12 C(=O)(C1Cc2cccc(Cl)c21)NC(C1CCN(C(=O)C(F)(F)CO)CC1)C O(NC(=O)C(C)(C)C1=CCN(C(=O)CCS(C)(=O)=O)C1)NC CC1C(NC(C2CCC(C)(C)O2)=O)CCN1C(=O)CC1CCN(S(C)(=O)=O)CC1 S(=O)(=O)(CCC(=O)Nc1ccc(NC(C2(C#N)CC3CC3C2)=O)cc1)N(C)C Cc1nncc(C(=O)NCc2cc(C(=O)NC(c3ccsc3)C)n[nH]2)c1C C12(NC(C3C(=C)C3)=O)CCCC1N(C(c1cc(N(C)C)ccn1)=O)CCC2 C1(NC(c2ccc(C)nc2)=O)CC2CC(NC(c3cnc(C4CC4)[nH]3)=O)CC12 CN1CCC2(C(=O)NCCOCCN(c3nccs3)C)CCCC12 Cc1cnc2n1CCCC2C(=O)NC(c1ccc2c(c1)OCCO2)CC(=O)N(C)C C(CC(=O)NC(C)CNC(=O)C(C)OC(C)=O)NC(=O)OC c1(OCC)ccc(C(=O)NC2CCC(N(C(=O)CCC(N)=O)C)C2)cc1OC c1(C(N2C(CC(=O)Nc3cccc(-c4ccncc4)c3)CC2)=O)ccccc1S N(C(=NCCCOC)NCc1nc(C(C)C)cs1)CC1CC1C(C)C C1(C(C)C)CN(C(C2CNC(=O)N2)=O)CCCN1C(=O)CCCC(N)=O N(C1COc2cccc(F)c21)C(=O)NC1CC1COc1cccc2ccccc12 C1(NC(COc2c(OC(C)C)cccc2)=O)CCN(C(c2cncs2)=O)CC1C C=CCC(CC(C)C)C(=O)NCC1(F)CC(CNC(=O)C(C)S(C)(=O)=O)C1 C1(CC(=O)NC(C=CC(=O)NC2(C(=O)OC)CCCC2)C)CC2C=CC1C2 C(N=c1[nH]ccn2nnnc12)c1cn(C2CCCN(C(C(CC#C)(C)C)=O)C2)nn1 c1(CC)[nH]nc(C(=O)NC2CC(CCC(=O)N3CC(N4CCC4)C3)C2)c1C c1(C2C(C(=O)OC)C2)ccc(CO)cc1.N1(Cc2ccco2)CCCC1C(=O)O N1(c2cc(C)c([N+](=O)[O-])cn2)CCC2(CCCCC2NC(=O)C(F)C2CCC2)C1 c1(C(=O)NC(C)CNC(c2cscc2Cl)=O)cc(=O)n2nccc2[nH]1 C1(C(=O)NCC(=O)OCC)CCN(C(C2(C)N=N2)=O)CC1 N1(C(c2c(CC)cno2)=O)CCOC(CN(C(=O)CCCF)C)C1 N12CCOCC(C)(C1)CNC2=O.C1(C)(CS(=O)(=O)NC(C)(C)C)CC2(CCC2)C1 N1(C(c2sc(C)c(C)c2C)=O)CCC2CN(C(=O)CCC(C)(F)F)C2C1 C1(C(N2CC(CC(C)NC(c3nccc(C)n3)=O)C2)=O)CCc2cnc(C)n2C1 CC(C)C(CCN(C(=O)CC1(N(C)C)CC1)C)NC(c1cncnc1)=O C1(C(n2ccnc2-c2ccc(F)cc2)C)CCN(CN2CCNCC2=O)CC1 n1(C(C(=O)NC)C)nnnc1CC(=O)OCc1ccn(C(F)F)n1 C1(NC(c2nc(C(C)=O)sc2)=O)CCC(C)N(C(c2nc(C)c(C)[nH]2)=O)C1 C#Cc1ccc(CCCC(=O)N2CCC(N(C(=O)CC(=C)C)CCO)C2)cc1 Cc1nc2c(NC3CN(C(=O)CC4CCc5ccccc5C4)C3)ncnc2s1 C(=O)(C(C#N)(CC)CC)NC(C(=O)NC(CCC=C)(C)C)Cc1ccco1 C(=O)(C(O)C(C)CC)N1CCC(N(C(C2CC(CC)C2)=O)CCOC)CC1 c1(C(=O)NCC2C=CC(NC(c3c(C)nn(C)c3C)=O)C2)cccc2c1OCC2 C#CCCCC(C)C(=O)N1CCN(CC(N2CCC(C)(C)CC2)=O)CC1 c1(C(N2CCCC2C(N2CCCC2)=O)C(=O)NC(CC)C)cnccc1C Cc1cccc(C(N2CC(NC(=O)Cc3cccc(O)c3)C(C)C2)=O)c1 c1(C(=O)NCC(C)(C(C)C)NC(C(C)SCC)=O)cccc([N+](=O)[O-])c1Cl C(c1cn[nH]c1)=C(C)C(N1CSCC1C(=O)NCC(O)C1CC1)=O Cc1ccc(F)c(C(N2CCC(O)(C(N3CC(C)OCC3C)=O)C2)=O)c1F c1(C2C(C)C2)nocc1C(=O)NC1CC(C)(CNC(=O)COCCF)C1 C(CC(C)C)(C(=O)NCCCF)N1CC(c2c(C)occ2)C1 CC1CC(NC(C2(c3ccc(F)cc3)CC2)=O)CN(C(=O)Cc2cccnc2)C1 C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1C(O)CCN(CC(=O)N(CC)CC)C1 CCC(CCC(=O)NC1(C)CC(O)C1)NC(=O)COCCCN(C)C C1(C(=O)Nc2cccc(C3CCC3)c2)C2CCC3C(C2)CC13 C1(C(=O)NC)CC(c2ccc(-c3cncc(S)c3)cc2)CC1O.C(=O)N(C)C(C)C C1(CNC(CC(=O)OC)=O)CN(C(C2(C)CNC(=O)C2)=O)CCC12CCOCC2 c1(C(=O)NC2CC(NC(CC3CC(OC)C3)=O)C2)ccc(C(F)F)cn1 N1(C(C2CC(SC)C2)=O)CCC(F)(CNC(=O)C(O)C(C)SC)CC1 c1(C(=O)NCCN(C)C(C2CC23CCSCC3)=O)ccc2c(c1)C(=O)CCS2 N1(C(c2ccc(SC)o2)=O)CCC2CC(C1)CN(C(=O)C(O)C1CCCC1)C2 c1(C(N2CCCN(C(c3n(C)nc(CC)c3Cl)=O)CC2)=O)cccc2sccc12 C12(CNC(=O)NC(CC=CC)CO)CCC(C(=O)O)(CC1)C2 c1(CNC(c2ncccc2F)=O)ccc(-c2ccncc2)cc1F C1(CNC(c2cn(CC)nn2)=O)CCC(NC(C2CCC3CCC23)=O)CC1 C1(NC(C(n2c(C)cc(C)n2)C)=O)CC2CC1N(C(C1CC(C)(O)C1)=O)C2 C(=O)(C1=NOC(C)C1)NCC1CCN(C(c2ccc(SC)s2)=O)C1 n1(C(C)C)ncc(C(N2CCOC(C(C)NC(=O)C=CCO)C2)=O)c1Br N1(C(Cn2ccc(C)cc2=O)=O)CCn2c(cc(CC(=O)O)c2C)C1 c1(CC(N2CCC2)=O)cc(=O)n(-c2ccccc2)[nH]1.c1(C(=O)O)ccccn1 c1(OCC)ccc(NC(=O)CN2CCN(Cc3cccnc3)CC2)cc1C C#CC1(O)CC(C(=O)NCCn2cc(C(=O)NC3C(C)(C)C3(F)F)cn2)C1 c1(C(=O)NC2CC(CC(N3CC(SCC)C3)=O)C2)ccc(C)o1 C1(NC(C2CC(=C)C2)=O)CC2CC1N(C(=O)C=Cc1cscn1)C2 C1(C(=O)NCC(CCCC)NC(c2cnc(C3CC3)[nH]2)=O)CC2CCC(C1)C2 C1(C(=O)NCC(C)C2CC2)CC(NC(=O)CC2CCCCC2)C1(C)C c1(NC(C)(CCCl)C(F)(F)F)cc(Br)c2c(c1)OCO2 C1(C(=O)NCC2(NC(C3CC4(CC4)C3)=O)CCCC2)(OC)CCC(C)C1 N1(C(C(=O)NC2C(COC)C2)=O)CC(CNC(=O)C(=O)N(C)C)C2(CC2)C1 c1(OC)cnnc(C(=O)NCCCOCCN(C)C(C2CCO2)=O)c1 c1(CNCCN2CCN(CCS(C(C)C)(=O)=O)CC2)cc([N+](=O)[O-])cn1C c1(C(=O)NC2CCCCCN(C(CCOC)=O)C2)cnn2c1CC(C)CC2 O=S(=O)(c1ccc(Br)cc1NCC1(CO)CC1c1ccccc1)NCC1(Br)CC1 N1(C(c2cnc(CC)[nH]2)=O)CCC(C2CC2)(CNC(=O)Cc2cncc(C)c2)C1 Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCCCC1CNC(=O)C=Cc1cc[nH]c1 C=C(C)c1cn(C(C)CNC(c2nc(C(F)(F)F)cs2)C2C(CC(C)(C)C)C2)nn1 C(N=c1ccc(I)c(F)[nH]1)c1c(Cl)cc(Cl)c(C(=O)OC(C)(C)C)c1Cl C1(O)(C(=O)NCCCOCCN(C(CCC)=O)C)CCc2ccccc2C1 CC1=CC(C)=NS(=O)(=O)N1CC(=O)Nc1nocc1Cl N1(C(c2cn(CC)nc2C)=O)CCC(CNC(=O)COCC(F)F)C(O)C1 n1(CC(=O)NC2CN(C(CNC(C)=O)=O)CC2C(F)F)ccc(O)nc1=O C1(CC)C(NC(=O)C#CC(C)(C)O)CCCN1C(c1cc(O)nn1C)=O c1(C(=O)NCC2C(NC(C(C)CC(F)F)=O)CCCC2)ccccc1[N+](=O)[O-] c1(C(=O)NCC(CCNC(C(CC)COC)=O)(C)C)ccc(C)c(F)c1F C(C)(C(C(=O)NCC(O)C(C)(C)O)C(C)C)NC(CCC#CC)=O N1(C(c2c(C)c[nH]n2)=O)CCC(N(C(=O)CCCc2cccs2)C)C2(CC2)C1 C1(c2n(-c3ccn(CC)n3)nc(CCN3CCCC3)n2)COc2ccccc2O1 C#Cc1ccccc1C(N1CC(C2(NC(c3cc(Cl)ccc3OC)=O)CC2)C1)=O c1(C(=O)NCCC(CNC(CCNC(CC(C)C)=O)=O)O)cc2c[nH]cnc-2n1 NS(=O)(=O)CC(=O)NC1CC(NC(C2CC23CCCC3)=O)C1 c1(OC)c(C(=O)NCCC(CNC(=O)C(O)CC2CC2)OCC)cccc1Cl N#Cc1ccc(CC(N2CC(O)(CCNC(=O)CCC3CNC(=O)N3)C2)=O)cc1 Cc1nc2cc(C(=O)N(CCCNC(=O)Cc3cc(F)ccc3Cl)C)cnc2s1 c1(C(=O)NC2(CO)CCN(C(CC=C(C)C)=O)C2)csc(=NC2CCCCC2)[nH]1 c1(OC)cc(C(=O)NCC(O)C(=O)NCCn2ccc(=O)cc2)n(C)n1 CC1CCCN(C(c2ccc(Cl)o2)=O)C1CCNC(c1cnc(C2CCC2)s1)=O C1(CNC(CNS(CC)(=O)=O)=O)CCC2CN(C(=O)CCn3ccnc3)CC12 C1(NC(C(C)CN2CCOCC2)=O)CN(C(=O)CC(F)F)Cc2nccn2C1 C(N=c1[nH]c(=NC2CC(n3cccn3)C2)c2[nH]ccc2[nH]1)C1OCC(C)(C)C1 C1(C(N2CCC(c3cn(CCC=C=C)nn3)C2)=O)Cc2ccncc2C1 CN1CCC(C(N2CCC(n3cc(CN(C)C)nn3)CC2)=O)C1c1ccccc1 N1(CCC)CCCCC1C(N1CC(CNC(=O)CCC2CCCC2)CC1C)=O Cc1cc(C)c(C(=O)NC2CC(CCNC(c3cc(C(C)C)[nH]n3)=O)C2)c(O)c1 n1(CC)cccc(NC(=O)N(c2ccc(Br)cc2F)C)c1=O C1(C)(CNC(c2ccc(CC)cn2)=O)CN(C(c2ccc(O)c(Cl)n2)=O)CCO1 c1(OC)ccnc(CNC(=NCC2CC2)NCC2(c3ccccc3)CC2)c1OC C12CSCN1C2=O.C(=O)(C(O)c1ccsc1)NCCCOC(=O)NC C1(CC(=O)NC(C(C)C)c2ncc[nH]2)CN(C(c2cnn(C)c2Cl)=O)CC1C C12(CNC(CNC(C)=O)=O)CCCC1(F)CN(C(=O)CN(C)C(N)=O)C2 Cc1nc(O)nc(S)c1C(N1CCC(C)C(NC(C2CCCC(C)C2)=O)C1)=O Cc1cc(I)c(F)cc1NC(c1n[nH]c2c1CN(C(c1cccc(F)c1)=O)C2)=O c1(CC)onc(C)c1C(=O)NC1CCCCC1CNC(c1nocc1Br)=O C(=O)(CC1=NN(C)C(=O)C1)N1CCC(OCCNC(c2c(C)nc(CO)o2)=O)C1 C(=O)(C1=NOC2(CCC2)C1)N1CCN(C(C(C)(C)C2CCCC2)=O)CC(O)C1 c1(C(N(C)Cc2cccc(CNC(=O)CNC(N)=O)c2)=O)nccc2c1CNC2=O C1(c2ccn(CCC)n2)(NC(C)CC)CCN(C(=O)OC(C)(C)C)CC1 CC(C(=O)NNC(=O)c1ccc(C#N)cc1)C(C)(C)C C#Cc1ccnc(C(=O)NC2C3CC2CN(C(c2ccncc2OC)=O)C3)c1 C1(OCC)CC(CNC(C2(n3ccnn3)CC2)=O)C12CCC2 Cc1sc(C(=O)NCC2CN(C(C3C(Cl)(Cl)C34CC4)=O)CCN2C)cc1[N+](=O)[O-] C1(NC(C(C)=O)=O)CCCC2CN(C(c3cc(Br)n[nH]3)=O)CC12 c1(C(C)NC(C2NCCN(C(C(CCCC)O)=O)C2)=O)cc2ccccc2s1 N1(C(c2cc(C)c(C)s2)=O)CCCOC(CNC(c2cccc(C(F)F)c2)=O)C1 c1(N(CCCC)C)nc(N2CCC(c3nc(=N)n(C)[nH]3)CC2)c2c(n1)CSC2 CC12CC(C(N3CCC(=CCOc4cccc(Cl)c4)CC3)=O)(C1)OC2C(F)(F)F n1(C2C(C(N3CC(F)CC3C(N3CCCC3)=O)=O)C2)cnc2ccccc12 C1(C(N2CCN(C(C3OC4CCC3CC4)=O)CC2)=O)CCC2(CCCC2)C1 N1(C(C2ON=C(C(C)C)C2)=O)Cc2nccn2CC(NC(C2C=CCC2)=O)C1 CN1CCC2CN(C(C3CC3NC(c3cc(O)no3)=O)=O)CC2C1 Cc1cc(C)n(C(C)C(=O)NCCCOCCNC(=O)CNC=O)n1 C1(C)(NC(c2cc(CNC(CC3C(C)=NNC3=O)=O)[nH]n2)=O)CC(C)(C)OC1=O N1(C(CC(CNC(c2coc(C(F)F)c2)=O)OC)=O)CCC(F)(F)CC1C N1(C(C2CC(C)C(=O)CC2)=O)CC2(CCN(C(C3(CO)CCC3)=O)CC2)C1 CC(C)CCC(O)C(=O)NCC(C)CN(C)C(C1CC(=O)NC(C)C1)=O N1(C(CSCC)=O)CCC2CCCC12CNC(=O)CS(=O)(=O)N(C)C C1(C(N(CC(CC)(F)F)C)=O)CC12CCN(C(c1cnc(C(C)C)o1)=O)C2 Cc1cc(C)c(C(=O)NC2(CN(C)C(c3ccc(C4CC4)s3)=O)CC2)cn1 N1(C(C(CO)NC(c2c(CC)ocn2)=O)=O)CCN(C)CC1C N1(C(C23CN(C(=O)OC(C)(C)C)C(C2)CO3)=O)CCC2(CCO2)CC1 C(=O)(CC(C(C)C)NC(=O)CC#N)NCC(CC)C c1(-c2n[nH]c(=NCCCNC(=O)OC(C)(C)C)s2)ccc(Cl)c2cccnc12 N1(C(C=C(C)c2cccs2)=O)CCN(C(C2CC3CCCC(C2)C3)=O)CC(O)C1 c1(C(c2nnnn2C(C)C)NC(CCC)CCO)c(Br)ccc2c1OCO2 CC1(C)CC(O)C(O)CN(C(CCC2CC2)C(=O)NC2CCC(F)(F)CC2)C1 C1(C(=O)OC)CCCC(C(=O)NC2CCCC(NC(c3nccnc3C)=O)C2)C1 N1(C(C2CC3N(C(CC(C)F)=O)C(CC3)C2)=O)CC2(CCOC(=O)N2)C1 O=C(NOCC1CCCO1)C1c2c[nH]nc2CN1C(=O)C1=NOC2(CCC2)C1 C1(NC(c2nc(C)sc2C)=O)CC2(CCN(C(=O)C(c3cccc(Cl)c3)C)C2)C1