SMILES N1(C(C2CC(CNC(c3cc(C)oc3)=O)OC2)=O)CCC(C)(F)CC1 c1(C(=O)NC(=O)CN)ccc2c(c1)CCC2.CC1CC(C)CN1C(=O)CC1CC1C c1(OC)ccnc(C(=O)NCC2(CO)CC2)c1C.C12CC(C)N(C1)C(=O)C2 C1(OC)CN(C(=O)CN2CCC(C)CC2)CC1NC(C1CCCN(C(C)C)C1)=O Cc1nn(C)nc1C(=O)NC1COCC1CNC(=O)CC(C)c1ccccc1 C1(O)(CNC(COCC#C)=O)CCCN(C(=O)C2=C(C)CCCC2)CC1 C(=O)(N=c1[nH]c(Cl)c(I)nc1Br)C1N(C(c2cccc(N)c2)=O)C2C(C1)C2 c1(C(=O)NC(C2CCCCN2C(c2cnc[nH]2)=O)C)ccc2nnnn2c1 C(=O)(C(C(C)O)NC(c1cnn(CCNC(c2ccncn2)=O)c1)=O)OC c1(NC(C2CCN(CCNC(=O)C(C3CCCCC3)O)CC2)=O)ccc(O)nn1 c1(CCC)cc(C(=O)NC2CCCC(CNC(C3CCCC(=O)O3)=O)C2)nn1C Cc1nccnc1C(=O)NCCn1cc(C(=O)NCC2COC(C)(C)C2)cn1 Cn1cnnc1C(=O)C(=O)NC1CCN(C(c2csnn2)=O)C1 N1(C(CS(=O)(=O)NC)=O)CC(C(=O)NC2(CO)CCC(C)C2)CC(C)C1 c1(C(N2CCCCC(Nc3c(C#N)c(Cl)ncn3)C2)=O)cc2cccc(F)c2o1 Cc1cc(-c2cncc(C(=O)Nc3nc(C4CC4)c(Br)s3)n2)cc(C)c1 C1(C(=O)OC)CC(C)N1C(=O)CCC1CCC1.C12(CC1C)C(=O)N2 CCC(CN=c1[nH]c(N(C)Cc2cc(Br)cn2C)nc2c1CCCC2)OC c1(OC)cc(Cl)ccc1C(C1CC1)NCC(=O)NCC1(C)CCC(C)C1 C1(O)(CC(=O)NC(CC)Cc2ccco2)CCCN(C(c2ccc(F)cc2)=O)C1 c1(C2CCN(C(CCSCCN(C)C)=O)C2)nnc2n1CCOC2 N1(C(CC2C(CC)C2)=O)CCn2ncc(CNC(c3cc(C(C)C)on3)=O)c2C1 C(=O)(CC(O)C(C)C)NC1(C(=O)NCc2ccn(CCC)n2)CC(F)(F)C1 c1(CC)ncc(C(=O)NC(C)(C)CNC(C2CC2CF)=O)s1 c1(C(=O)NCCN(C(c2c(CC)c(F)ccc2)=O)C2CC2)cc2ccccn2n1 C1(NC(c2cn(CCC(C)C)nn2)=O)CN(C(=O)C=Cc2ccoc2)CC12CC2 c1(-c2cn(C3C(NC(=O)OC(C)(C)C)COC3)nn2)cncc(C(F)(F)F)c1 c1(C(=O)NCCCC2CCN(C(C(OC)OC)=O)CC2)cn2ncccc2n1 Cc1csc2c(N3CC(O)(CCNC(C4CC(F)(F)C4)=O)C3)ncnc12 N1(C(CCC)=O)CCC(NC(c2nccnc2Cl)=O)C(F)C1 O=C(CCCc1cccs1)NC(C1CCCCC1)C(=O)NCc1ccon1 CC1(C)CC(NC(c2ccc(C(F)F)s2)=O)CN(C(c2c(Cl)cccc2Cl)=O)C1 N1(C(C2=C(C)OCCC2)=O)CC2CCCCC2(NC(C2COCCO2)=O)C1 c1(N2C(C)CC(CNC(C3CC(O)C3)=O)C2)ncc(F)c(-c2ccsc2)n1 C1(C(N2CCCC(CC(=O)NCCc3ncon3)C2)=O)CCCC1C1CC1 N1(C(c2c(C(C)C)nns2)=O)CCCN(C(=O)C2=COCC2)CC1 CCC(C)(COC)C(=O)OCCOCc1cc(O)nc(OC)n1 c1(NC(CCN(C(=O)C(F)CC2CCC2)C)=O)cnc2ccnn2c1 C1(C(N(C2CCC2O)C)=O)CCCN(C(c2cnnc(O)c2)=O)C1 CS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(C34CCC3C4)=O)C2)c1 N1(C(COC(CC)C)=O)CCC2CCN(C(c3c(O)cc(F)cc3F)=O)CC2C1 N1(C(C)C)CCC(CNC(c2ccc(-c3cnn(C)c3)s2)=O)C1 c1(NC)cc([N+](=O)[O-])ccc1CN1CC2(CC2C(=O)NSc2ccc(Br)cc2F)C1 N12CCC(O)(CC1)C(=O)NC(CC)C2=O.C(Cc1ccccc1)(C(=O)OC)NC C1(C(N2CC3C(CNC(Cc4cc(C)no4)=O)(C3)C2)=O)CC2(C1)CC(C)C2 c1(CNCc2cn(-c3c(C)ccnc3)nn2)ccc2nnnn2c1 N1(C(C(=O)NC(C)C)=O)CCC(NC(c2scnc2C(F)(F)F)=O)C(F)C1 Nc1cc(C(=O)NCC2(NC(=O)CC3(O)CCC3)CC2)cc(F)c1 C1(CC(=O)NC2(C(N)=O)CC2)CC(=O)NC1=O.c12conc1C(C)CNC2=O N1(C(CNS(NC)(=O)=O)=O)CC(CNC(=O)Cc2nonc2C)N2CCC1C2 c1(OC)ccc(Cl)c(C(N2CC(NC(c3nc(C(N)=O)co3)=O)C3(CC3)C2)=O)n1 c1(OC(F)F)cc(CCNc2ccnc(OC)c2)cc(F)c1OC.CO CC1(C)C(NC2CCC23CCCC3)CC1O N1(C(C2(CC)CCCC2O)=O)CC2(CC(CC(=O)NC3CCCSC3)C2)C1 C(C(CC(=O)NC1(CCN2CCCCC2)CC1)NC(=O)Cc1cccn1C)OC CC1=NOC(CC(N2CCCC2C2(C(=O)NCCN3CC4CC4C3)CC2)=O)C1 C1(C(=O)NCC2(F)CCN(C(CP(C)(C)=O)=O)C2)CC1C1(C)COC1 N1(CC(=O)NC(C)Cn2cc(COC3CCOC3)nn2)CCNC(=O)C1C [SH](=O)(=O)c1cnc2ccnn2c1.CC1Cc2cscc2CN1C(=O)CCCCCC#N C12CCN(CC1(C)C)C(=O)c1[nH]ccc1CNC2=O.C1(CC#C)(OC)CC1 N1(C(CC)=O)CCCC(C(N2CCC3C(NC(c4ncn(CC)n4)=O)C23)=O)C1 c1(C(=O)NC2C(NC(C=CCCC)=O)C2)cnn(-c2ccc(F)cc2)c1C.C(=O)OC CC1CC(NC(C2(C)CCN(C)C2=O)=O)CCN1C(=O)Cc1cc(Cl)cc(Cl)c1 C(=O)(C(CCCCN)CC(F)(F)F)NCCC(N1CC(c2cc(C)on2)C1)=O C(C(N=c1[nH]c(C2CCOCC2)nc(Cl)c1C)C(C)C)NC(C(CC)C(C)O)=O N1(C(=O)OC(C)(C)C)CCCC2(CCN(CC)C2)C1.[nH]1nc(C2CC2)cc1CSCC C1(NC2CCC(C(=O)O)C2)CC2COCC2C1.c12nc(cs1)CC(=O)N2C(C)=O c1(CNC(C2CCCN(C(C(C)SCC)=O)C2)=O)c(OC)cc(Cl)cc1F C(CCN=C(NCCSc1ccc(F)cc1)N1CCC(C(F)(F)F)(CO)C1)SC Cc1ccc(N2CCCC2NC(=O)NCCCN2CCC(O)C2)cc1 N1(C(C(=C)C(F)(F)F)=O)CC2CC(C1)CN(Cc1c(Cl)[nH]c3ccccc13)C2 C(=O)(C(C#N)C(C)(C)C)NC(C)(C)CCNC(=O)Cc1cncc(O)c1 N1(C(c2c(C)coc2)=O)CC(C)N(C(c2cc(Br)c(Cl)cc2C)=O)CC1C C(C1=NOC2CCCC12)n1cc(C2(CO)CN(C(C(C(C)C)CC3CC3)=O)C2)nn1 c1(C(N(C2CCN(C(=O)CC3CCC4CC34)C2)C)=O)ccnn1CCF CC1CCN(C(C2CCC(NC(C3CCCC4(CC4)C3)=O)C2)=O)CCO1 C1(C2CCN(C(=O)C(C)(C)C(C)O)CC2)(NC(CCCOC)=O)CC1 N1(C(CC(CCC)NC(c2ncn(C)n2)=O)=O)CC2CCN(C(C)=O)CC12 C1(C(=O)NCc2occ(C(N3CCC(CC)(OC)C3)=O)n2)CC2COCC2C1 N1(CCCS(C)=O)CCN(Cc2ccc(C(C)(F)F)cn2)CC1 N#CC1CN(C(c2cc(Br)cnc2Br)=O)CCN1C(=O)C=Cc1cccc(F)c1 C1(NC(C2C(C)C2)=O)CC(F)(CCN2CCOCC2)C1.n1(C)cc(C(C)N)nn1 C#Cc1cc(C(N2CCC(CCNC(=O)C(C)CCC)C2)=O)cc(N)c1 C(=O)(CC(C)(C)C(=O)NCC1(NC(=O)CS(N)(=O)=O)CCOCC1)OCC c1(CC(C(=O)NCC(N(C(COCCCC)=O)C)C2CC2)O)ccc(Cl)cc1 C1(CCC)(NC(c2ncccc2C(F)F)=O)CCCN(C(C2CCOC2)=O)C1 C1(C(N2CC(O)(CNC(CC3C(C)CCO3)=O)C2)=O)CC(=O)NC(=O)C1 C1(NC(C2C(C(C)NC(C(CC)CN(C)C)=O)C2)=O)CC2(CCCCO2)C1 CCC(C)CCCC(=O)NCCC1CCCCN1C(c1cccc(C#N)c1)=O Cc1ccc2c(C(=O)NC3CCCN(c4ncnc5ccsc45)C3)cn(C)c2c1 C=Cc1cc(C(=O)NCCCN(C(c2cc(CSC)on2)=O)C2CC2)cc(F)c1 CC1CCCC(C)N(C(c2conc2CNC(=O)C(C)n2cccn2)=O)C1 C1(C(=O)NC2(C(=O)NCCc3cc(C)ncc3)CC(O)C2)CCCC(C)CC1 c1(C(N2C(CNC(C(CSC)O)=O)C(C)(C)CC2)=O)cccc2c1COC2 c1(C(=O)NC(CC2CN(C(c3ccc(C(C)C)o3)=O)C2)C)cc(O)nc(O)n1 CC(O)C(=O)NNC(=O)NCCC(c1cccc(F)c1)C C(=O)(C(C)(CSC)NC(c1cc(OC)n(C)n1)=O)NCC(CC)C#N N1(C(C(C(C)CC)N(C(C=CC)=O)C)=O)C2CCC1CC1(CC1)C2 c1(OC)ccc(F)c(N)c1C(=O)NC(c1ccc(-n2cncn2)c(F)c1)C C1(CC(=O)NC(CNC(C2(SCC)CC2)=O)C(C)C)CCCCCO1 C1(NC(C2C(C(=O)OC)C2)=O)C2COCC1CN(C(c1n[nH]cc1C)=O)C2 C=CC1CN(C(C2C3CC4C(C3)C24)=O)CC1NC(=O)C(C)CC(N)=O CC1(CNC(C2CC(NC(c3ccc(O)cn3)=O)CCO2)=O)CC=CCC1 CC(C)=C=CC(=O)N(CCC(c1cccs1)NC(=O)CC(C)C)C C1(C(C)O)CCC(NC(C2CC2F)=O)CC1.c12cn(nn1)C1CC(C1)OC2 CCC(CC)(CO)C(=O)NCCC1CN(C(c2cc(Br)n(C)c2)=O)C1 CC(C)(C)C(C(=O)Nc1cccc(NC(=O)C2=CCCS2)c1)C1CCCCC1 C1(C(=O)NCc2c(CCNC(=O)CC3CCCS3)ocn2)CCCN1C=O N1(C(=O)C=Cc2cccnc2)CCN(C(c2cc(CC3CC3)on2)=O)C2CCC12 C(=O)(C(C)CCCCCC)N1CC(C(N2CC(C#C)(F)C2)=O)C(C)(C)C1 c1(CNC(c2n(CCCOC)nnn2)CCCSC)ccnc(Cl)c1Cl C(=O)(C(=O)C(C)(C)C)NC(CCC)C(=O)NCC(C)N(C)C c1(OC)c(Cl)cc(C(=O)NC23CC(C2)N(C(c2nc(=N)cc[nH]2)=O)C3)nc1Cl Cn1cnc(C(N2CC(O)(C(C)(C)CNC(C3C=CCCC3)=O)C2)=O)c1 CCCC(CCCNC(c1cc(CC)nn1C)=O)NC(c1coc(C(N)=O)c1)=O N1(C(C)=O)CCCC1(C)C(=O)NCC1(O)CCN(C(=O)CCCC2CC2)C1 C#Cc1c[nH]nc1C(=O)NCC1CC(F)CN1C(c1ccoc1Cl)=O c1(C(=O)NC(CC=C)CNC(c2ncn(CC)n2)=O)ccc(C2CC2)cc1C c1(CC)ccc(C(=O)NC2CCC(C)N(C(c3cc[nH]n3)=O)C2)cc1CC N1(C(CCC2CC(NC(Cc3c(C)nn(C)c3)=O)C2)=O)C2CCC1CC(C)C2 c1(N2C(CNC(C(C(CC)O)C)=O)CCCC2)nc2c(F)cc(Cl)cc2s1 C(CC(CC)C(=O)NCC(O)CC(=O)NC(C)C(C)C(=O)OC)=CC C(=O)(CCCC(C)(C)C)N1CC(C(=O)NCCCC(=C)Cl)C(C)C1 n1(CC)cc(C(=O)NC23CC(C2)N(C(=O)CN2CC(C)(C)C2)C3)c(C)n1 c1(N2CC(O)(C(C)NC(c3cnc(-c4ccco4)s3)=O)C2)ncc(Cl)cn1 C1(N(C(c2cc(CCO)on2)=O)CC)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 c1(C(N2CCN(C(C=C(C)c3cccs3)=O)C3C2C3)=O)ccc(S(N)(=O)=O)nc1 C(=O)(C(C(C)(C)C)c1ccccc1)N1CCC(N(C(c2c(C)snn2)=O)CCO)C1 CCCC(CCCNC(C1CCCO1)=O)NC(C1(N(C)C)CCCCC1)=O CC1(C)CCCOC1C(=O)NC(Cn1cncn1)C(=O)NCc1ncc[nH]1 CCC(CC)C(c1nnnn1Cc1ccco1)NC1CC1C(C)(C)C CC1OC2(CNC(=O)COC3CCCC(C)C3)CC1(NC(C1CC1(F)F)=O)C2 CN1C(C(N)=O)CCC1C(N1CCOC(CNC(C2(C(C)(C)C)CCC2)=O)C1)=O C1(CNC(CC(C)(C)NC(=O)CCNC(=O)CO)=O)CC2(CCCO2)C1 c1(C(=O)OCCN2CCN(C(c3c(OC)ccs3)=O)CC2)cc(F)c(Cl)c(Cl)c1 C#CCC(CC(=O)N(C(C)C(=O)N(C)C)C)NC(=O)C(SC)SC c1(CC(C)C(=O)NCC(O)CCNC(=O)CN(C)S(N)(=O)=O)ccccc1Cl CC1CN(C(c2c[nH]nc2-c2ccco2)=O)CCN1C(=O)CC1CC(=O)C1 c1(C(=O)NC2C(NC(C3(CC(=O)OC)CC3)=O)CCCC2)ccc(S(N)(=O)=O)o1 c1(C(=O)NCCN(CC(O)CO)CCCC)nc(C)oc1C(=O)OC C1(C(N2CC(O)CC(NC(C(CCOC)(C)C)=O)C2)=O)CCc2c[nH]nc2C1 c1(C(N2CC(CC(C)NC(=O)C(F)=C3CCC3)C2)=O)cc2ccccc2s1 c1(NC(c2scc(C(=O)O)n2)=O)ccc(C2=NOC(CN3CCCC3)C2)c(F)c1 c1(NC(=O)NCC2CCCOCC2)cc(CC23CC(C2)C3)ccc1F C12(C(N3CCCC(C)(CNC(C4CC4F)=O)C3)=O)CC3CC(C1)CC(F)(C3)C2 C(CCCC(=O)NCCc1ccon1)NC(C(C)c1cc[nH]n1)=O N1(Cc2cc(C(=O)OC)c(Br)cc2)CC2CN(C(c3cccc(F)n3)=O)CC12 N1(C(C(CC)CO)=O)CCC(C2CCN(C(=O)C(C3CCOCC3)C)CC2)CC1 c1(NC(C2C(NCc3cn(CC)nc3)C2)=O)cc(F)ccc1C c1(C(=O)NC(C)CCNC(c2n[nH]c(C3CC3)n2)=O)cncc2cccnc12 C(CC(N)=O)(C(=O)N1CCC(C)(C)CC1)NC(c1c(OC)noc1C)=O C(=O)(CCCCO)NC(CC(C)NC(C(C)OCC(C)C)=O)C C1(C(N(CC(=O)O)CCO)=O)C2CC(c3ccccc3)C1C2 c1(OC)ncc(C(=O)OC2CCCC2n2cc(-c3cncc(N)c3)nn2)cc1C C=CCCCC(=O)N1CCCC1CCNC(C1(OC)CC(C)C1)=O Cc1ccc(Br)cc1NC(N(CCO)Cc1ccc(C)c(Br)c1)=O N1(C(C2(F)CCN(C(COc3cn(C)nc3)=O)C2)=O)CC(C#N)C2(CCC2)C1 C(=O)(C#CC1(C)COC1)N1CC(N2CCC(NC(C3C(C)OC(=O)N3)=O)CC2)C1 C1(CNC(C=C(CC)CC)=O)CC2(CCC2)CN1C(c1ncc(CC)cn1)=O Nc1ncc(C(N2CCN(C(=O)C=CC3CCC3)C(C3CC3)C2)=O)cc1Br N1(C(c2cc(=N)[nH]cc2)=O)CCC2(CCN(C(C3CCCS(=O)(=O)C3)=O)C2)C1 C(=O)(C#CC1CC(F)(F)C1)NCC1C(NC(CC(C(C)C)C)=O)COC1 C1(CCC)(NC(=O)CCc2cc(C)[nH]n2)CCCN(C(=O)CS(=O)(=O)CC)C1 c1(OC)cc(F)c(C(N2CCOC(CNC(=O)CC3COCCO3)C2)=O)cc1N C1(C(=O)NCC(CC=C)O)CC(C)(C)CN1C(c1ccnc(O)c1F)=O c1(CC)ccc(C(C)C(=O)NC2C3CC2N(C(C2CCOC(=O)N2)=O)C3)cc1 C1(NC(C2CCCC2)=O)COC2(CCCN(C(=O)COc3cncc(Cl)n3)C2)C1 CCCC(C)(O)C(=O)NC1CC(C)(NC(C2CCC2(C)C)=O)C1 c1(C(N2CCC(C)C(NC(=O)CN3CCNC(=O)C3)C2)=O)cccc2ccoc12 CCCCC(CNC(C1OCCCO1)=O)NC(c1ccc(=O)oc1)=O C1(CC(=O)NCC(C)(O)C2CCCC2)C2CN(C(c3csc(Cl)c3)=O)CC12 CC(C)CC(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(=O)NC2CC(N3CCC3)C2)C1 N1(C(C)C)CCCC1C(=O)NCCCCNC(=O)Cc1cc(C(F)(F)F)n[nH]1 c1(C(N2CCOCC(NC(C(CC)(C)C)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 c1(OC(C(=O)NCCN(C(=O)CC(C)n2cccc2)CCC)C)ccccc1F N=c1[nH]cnc2c(C(N3CCCC(NC(=O)C(F)=C4CCC4)CCC3)=O)cnn12 c1(CC(CC)NC2CNCCC2C(F)(F)F)cc(Br)cc(Br)c1 Cc1c(C(=O)NC(C)(CO)C(=O)NC2CCN(CCCO)C2)ccn1C c1(NC2(CNC(=O)CCN3CCCS3(=O)=O)CC23CCC3)ncc2ccnc-2[nH]1 N1(C(CSc2n(C)ccn2)=O)CCC(CO)(CNC(=O)CC2CCSC2)C1 C(=O)(CCN=C(NCC(=O)N(C)C)NC(c1cnn(C)c1)C1CCCC1O)NC C#Cc1ccc(NC(C2CCC(CNC(c3coc(CO)c3)=O)O2)=O)cc1 c1(C(Cn2ccc(C)n2)NC(=O)CCNC(=O)CCl)ccccc1Br CC(C)(CC(=O)NCC1CCC1NC(c1cc(F)ccc1F)=O)CC(F)(F)F C(CC(C)C)(C(=O)N1CCC(OC)CC1)ONC(c1c(CC)n[nH]c1)=O N1(C(c2c(C)ncs2)=O)CC(NC(=O)C(C)CC(C)(C)C)CC(C)(C)C1 CC(C)(C#CC(=O)NCc1nc(C(C)(C)C)ns1)CNC(=O)OC(C)(C)C C1(NC(c2cccc(OCCC#C)c2)c2nnnn2C2CC2)CCN(C)C(C)C1 c1(C(=O)NC2(C=C)CCC2)c(-c2cccc(Br)c2)noc1C(C)C N1(C(c2n(CCC)ncc2)=O)CCCC(NC(c2cncc(C(C)(C)C)c2)=O)C1 C1(C(N2CC(O)(C(C)NC(c3c(C)cc(F)nc3)=O)C2)=O)CC(C)CC(C)(C)C1 C12(CNC(C3N(CC)CCCC3)=O)CCC(CC1)CN2C(=O)C(C#N)C(C)C Cc1cn2cc(C(=O)NCCc3nn(C)c(C)c3Br)sc2n1 C#CCCN=C(NCc1ccc(OC)c(S(N)(=O)=O)c1)NC1CCOc2cc(Cl)ccc21 C1(CC)CC(C(=O)NC2CN(C(C3CCOC3C)=O)CC2C)CCO1 C1(C(=O)NC2C(COC)CCC2)CC(O)CN1C(=O)CCCc1ccsc1 C1(C(N2CC(CN(C)C(C3CCCS3)=O)OCC2)=O)CC(C)(C)CCO1 CC(C)(CNC(C1(C)CC2CCC1O2)=O)CC(=O)NCCc1ccnc(O)c1 C12(C(=O)NC(C=C)C3CC3)CC(C)(C1)OC21CCC1 CC1=C(CNC(C2CC(NC(c3ccoc3)=O)C(O)C2)=O)COCC1 C1(NC(C2CC3CC3C2)=O)CCCCN(C(c2cc(Br)cnc2O)=O)C1 C1(C(=O)NC(COC)C2(C)CC2)CCCN(C(=O)CC2(CO)CCCCC2)C1 N1(C(c2c(C)nc(C3CCC3)o2)=O)CCN(C(=O)Cc2occc2C)C(CO)C1 CC1(C)COC(C(=O)NCC(C2CC2)NC(=O)CCN2CCOC2=O)C1 N1(C(c2c(CC)n(C)nc2)=O)CCN(C(=O)COCCN(C)C)C2CC12 c1(C(=O)OC(C2CCCCC2C)C)cc2c(cc1F)NCCC2 C1(C(=O)NC(CC=C)CC(F)F)N(C(=O)CCc2cc(C)on2)CCCC1(C)C N1(CC(=O)N(C(C2CC(Cc3ccccc3)=NO2)=O)C2CC2)CC2C(C1)C2(F)F C1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)O)CNC(=O)C(C)(C)C1 C(=O)(C(C(C)CC)N(C)C(c1ccncc1O)=O)NC(C#C)C(C)(C)C CCC(C#N)C(=O)N(CCN(C(=O)CCOC)C)C N1(C(C(CNC(c2ccc(C#N)s2)=O)CC2CC2)=O)CC2COCC(C2)C1 N1(C(C(C)(C)C2CC2)=O)CCN(C(=O)CC2CCOCC2)C(C(C2CC2)C2CC2)C1 CCC(C)CC(C(=O)NC1(CCF)CCOCC1)NC(=O)CC1CCCCCC1 C1(NC(C2(COC)CC2)=O)CCOCC1C(=O)NCc1ncn(C)n1 N1(C(C2C(C)C2C)=O)CCCC2(CCCN2C(c2ccsc2Cl)=O)C1 N1(C(c2cc(CCC)n(C3CC3)n2)=O)CCC2CN(C(C3CC3(C)C)=O)CCC12 c1(C(N2C(CC)CN(C(c3cocn3)=O)CC2)=O)cc(F)c(F)cc1OC C1(C(=O)NCC(C)(CO)NC(c2cnn(C)c2C#N)=O)(OC)CCCC(C)(C)C1 C(=O)(C1CCc2cccc(F)c21)NCC1(O)CCCN(C(C(CC)COC)=O)C1 c1(OC)ccccc1C(=O)NCC(=O)NC1CC1CNC(C1CC2C=CC1C2)=O CC1CN(C(c2nscc2Br)=O)CCCN1C(=O)CCCc1ccccn1 n1(C(C)NCC(O)CN(C(=O)CCc2ncc(C(C)(C)C)o2)C)cnc(C)c1 c1(C(N2CC(C(C(=O)NCc3ccco3)OC)C2)=O)cncc(F)c1C C(=O)(C1CCCc2ncnn21)NCCNC(=O)Cc1csc(-c2ccoc2)n1 C=CC(O)C(C)(C)C(=O)N1CCCC(C)(NC(=O)C(C)C(=O)OC(C)(C)C)C1 c1(OC(CC)C(=O)NCC2CC(NC(=O)CCN3CCCC3)C2)ccccc1F CC1CN(C(=O)Cc2cscn2)CCN1C(c1ccc(-n2nccc2C)cc1)=O C12(C(=O)NC(c3ccncc3)CNC(CSC)=O)CC(c3ccccc3)(C1)C2 C(C(C)(C(=O)NCC(C)(Cn1cccn1)NC(C1CCCN(C)C1)=O)OC)OC c1(N(C(=O)C(c2ccccc2)=O)C2CC2)ccccc1-n1nnc(-c2ccco2)n1 CN1C(=O)CSC1=CC(=O)N1CCC(NC(c2ccnc3cccnc23)=O)C1 C1(CNC(C2C(F)(C(=O)OC)C2)=O)COCCN1C(c1ccoc1C1CC1)=O C1(NC(CCCOCC=C)=O)CCC(NC(=O)C(C)(CO)NC(C)=O)CC1 Cc1cnc(C)c(NC(=O)C(O)C2CN(C(C3CCCC(=O)N3)=O)C2)c1 CC12CN(C(c3cnc(-c4ccoc4)[nH]c3=N)=O)CC1CS(=O)C2 C1(CCN(C(C2CCN(CCC)C2)=O)C)CCN(CCNC(C)=O)CC1 C=CC(CCC)CC(=O)N1CC2(C)CC1(C(=O)NC1CC(C(=O)OCC)C1)C2 N1(C(C(C)OC)=O)CC2(NC(C3CC3c3csc(Br)c3)=O)CCC1CC2 C1(CN(C(=O)CCSc2ccc(C)cc2)CC)CCCN(C(=O)CS(C)(=O)=O)C1 N1(C(CCC=C(C)C)=O)CCC2(CC1)CC2C(=O)NCCc1cccs1 C1(N(C(=O)CCC2CCCO2)CCC2CCC2)CCCN(Cc2ccccc2)CC1 C1(CC(=O)NCC(C)(C)NC(CC2CCC(C)CO2)=O)CCCC2(CCC2)O1 c1(C(=O)NC(C)CCN(C(=O)CC(O)C2CCCC2)C)ccc(P(C)(C)=O)cn1 C1(C)(CNC(c2c(C)cno2)=O)CCCN(C(C2(n3cncn3)CC2)=O)C1 C12(c3n(C)ncc3)CCC(C1)C2C(N1CCCC1CCNC(C1CC1CF)=O)=O c12ncccc1C(=O)N1CCC(C1)S2.C(=O)(C1=CCCS1)N(C(C)C)C C(C(=O)NCC(C)(O)CNC(c1ncnn1CC)=O)(C(C)C)OCC CC(C)CC(C(=O)NCC1C=CCOC1)NC(c1cnc(S)nc1)=O C1(NC(C2(F)CC2)=O)CCCN(C(=O)CCOC2CC2)C1 CC1CC(C(=O)NC2CCCCCC2NC(c2cn(C)nc2C(C)(C)C)=O)=NO1 CN1C(=O)CCC1(C)CNC(C1(CO)CCN(C(C2CCCC2C2CC2)=O)C1)=O c1(C(=O)NC(CC)C(=O)N(C2CCCN(CC)C2)CC)cccc(N)c1 C(=O)(CCCS(C)(=O)=O)NCCC(C)CCNC(=O)CCc1ccnc(Cl)c1 CCC(CC)CCCC(=O)NCC1(C)CCCN1C(=O)Cc1c[nH]ccc1=O N1(C(c2cc(SC)oc2)=O)CCC(O)CC1C(=O)NCC1=CCCC1 C1(O)(C(=O)NCC2(C(=O)NCC(=C)CC(F)(F)F)CC(=C)C2)CCOCC1 C12(C(=O)NC(CC)C(=O)OC)CCN(CC1)CC2.C1(Cn2ccnn2)C(=O)N1 C=CCC(C(=O)NC1COC(C(C)C)C1)NC(c1ccc(O)cn1)=O C(=O)(C1(C)CCn2ccnc21)NCC(CC)NC(C1(F)CCC1)=O N(C1CCCOc2ccc(Br)cc21)C(=O)NCC1CN(C)CC1C(F)(F)F C1(C(=O)OC)CCS(=O)(=O)CCN1C(=O)CSCC(=O)Nc1c(Cl)cccc1Cl C1(NC(C2CN(S(N)(=O)=O)C2)=O)CC2CC(C1)N(C(=O)CS)C2.c1(CC)cccs1 C1(C(=O)NC(C(=O)NC(C(CCC)O)CO)CCOCCO)CCC2(CCC2)O1 C1(CC(=O)NCC(C)NC(c2cc(O)ccc2Br)=O)CCCC(C)(C)O1 c1(C(C)C)ccc(C(N2CC(O)(CNC(c3ccc(-c4ccco4)s3)=O)C2)=O)o1 CN1CCN(C(C2(C)C=CCC2)=O)C(CNC(c2cn3c(n2)SCC3)=O)C1 c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)CC3CC3)C2)c[nH]c2ccc(F)cc12 c1(OCC)cc2c(cc1CN(C1(C(=O)O)CCSCC1)C1CC1)OC(C)C2 c1(C(C(=O)NC23CC(CNC(C4C(C#C)C4)=O)(C2)C3)O)ccc(C2CC2)cc1 c1(C(N2CCC(NC(COCCC(C)C)=O)C2C2CC2)=O)ccc2ccsc2c1 C1(C(=O)NC2CCOCC2NC(c2cc(O)nc(O)c2)=O)(OC)CCC(C)CC1 C(CN=C(NCc1cn(C)nc1Br)NC1CC1)OC(=O)NC c1(OCC)cc2ccccc2cc1C(N1CC(CNC(=O)CC(F)(F)F)C1)=O c1(C(=O)NCCC2CC(C)C2)ccc(S(=O)(=O)N2CCC(C(F)(F)F)C2C)c(Cl)c1 C(=O)(CCCCCc1cccs1)NCCC1(C(=O)OC)CCC1 c1(C(=O)NCCCCN(C)C(c2cnc(O)n2C)=O)ccc(Cl)c(C(F)F)c1 N1(C(C(C)c2ccsc2)=O)CCN(C)CC1C(=O)NCCCNC(N)=O N1(C(C2CCC(NC(C3ON=C(C)C3)=O)C2)=O)CCCC(C)(C(=O)O)C1 CCCCC(CC(=O)O)NC(C1CCCN1Cc1ccccc1)=O C1(C(=O)NC2(CNC(c3nc(OCC)oc3)=O)CC2)OC2CCC1C2 C1(=O)C(CC(=O)OC(C)(C)C)N1.C(C(C)C)N(C(C)C)CCO.C(C)(=O)O c1(C(N2C(CNC(C(CC)(C)OC)=O)C=CC2)=O)cccc(S(=O)(=O)C2CC2)c1 c1(C(=O)NCCC2(O)CN(C(C(CC=C)C)=O)C2)cccc2oc(=N)[nH]c12 C12(NC(=O)NCC(=O)OC)CC(CNC(=O)C(C)n3cccn3)(C1)C2 C1(CN(CC(C)NC(=O)CCn2cccn2)C)CCC1CN C(C(F)(C(=O)N1CC2CC1CC2CF)C(C)C)NC(Cc1c(C)n(C)cn1)=O C(C(CC(=O)N1CCOC(CO)C1)C1CC1)N(C(CC1(CCN=[N+]=[N-])CC1)=O)CC N1(C(=O)Nc2cc(C)sc2Cl)C2CCC(C2)C1c1ccccc1C(=O)OC(C)C C(C(C(C)(C)C)NC(c1cccnc1CO)=O)NC(CC(C)OC)=O C1(CN(C(c2ccc(C)o2)=O)CC)CCCN(C(=O)CCC(C)C)C1 C1(NC(c2c(COC)ccs2)=O)CC2CCC1N(C(=O)CCS(C)=O)C2 C1(NC(c2c(CC)cc[nH]2)=O)C2CCC1N(C(=O)Cc1cnc[nH]1)C2 C1(OCC(=O)NC(C)(C)CCNC(c2nc[nH]c2C(C)(C)C)=O)CCCCCC1 N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CNC(=O)CCC(C)C Cc1[nH]nc(CNC23CN(C(=O)CNC(N4CCOCC4)=O)C(C2)C3)c1C N1(C(C2(C)CCC2)=O)CCC(C2(NC(c3sc(Cl)cc3Br)=O)CC2)C1 C1(CC)CCN(C(C2CCC(C)O2)=O)C(C(N2CCC(CCCO)C2)=O)C1 O=C(CC(CC1CC1)NC(C1CC12CCCCC2)=O)NOCCC(F)(F)F c1(C(=O)NCCN(C(=O)CCCS(N)(=O)=O)CCOC)cc2c(cn1)OCCO2 C1(OCC)CCCC1NC(c1c[nH]nc1CNC(=O)CCc1ccncc1)=O c1(C(N2C(CC3(NC(=O)CC4CC4)CC3)CCC2)=O)n[nH]c(C2CC2)c1Br C1(N(C(CCOC)=O)C)CCCN(C(C2CCOC2(C)C)=O)C1 C1(CNC(c2cc(C)nc(C)c2)=O)CCC2CN(C(=O)C#CC3(C)COC3)CC12 c1(C(=O)NC(CNC(=O)C=Cc2ccccc2Cl)CO)c[nH]c2cccnc12 C1(C(N2CCC(C)(N(C)C)C2)C(=O)NCCC)CCC(C(=O)NCC)CC1 NS(=O)(=O)c1ccc(C(N2CC(NC(=O)C(F)(F)c3cncs3)CC(F)C2)=O)o1 c1(CN2CCC3(C(NC(C4CC(=C)C4)=O)C3)CC2)cn(C)c2ncccc12 C(=O)(C(C(C)(C)C)C1CCC1)N1CC(N(C(c2cnc(CC(C)C)s2)=O)C)C1 c1(C(=O)NCC2C(OCC)CN(C(c3cc(Cl)no3)=O)C2)c(Cl)ccc(C)c1O N1(C(C(C(CCC)NC(c2nnccc2C)=O)O)=O)CCCC(N=[N+]=[N-])CC1 N1(Cc2cn(C(C)(C)C)nc2)CC=CC2COCC12 c1(CC)cc(C(=O)NC2C=CC(CNc3nccc(C(F)(F)F)n3)C2)sc1C c12ccnn(c1=O)CCNC(=O)NCC(C)NC(=O)C2.C(F)(CNCC(C)C)=CC CCC(CCCC(=O)N1CC2C3CCC(C3)C12)NC(=O)Cc1ccn(CC)n1 c1(C(=O)OC)cccc(CNC(C)(C)CCCF)c1Br N1(C(C)C)CCCC(C(=O)NC2C3CCN(C(c4cc(C5(O)COC5)on4)=O)C23)C1 N1(C(c2c(C)cns2)=O)CC2CCCC2(C(=O)NCC2=NOC(C)C2)C1 C1(CC(=O)N(C(CCCCC)c2cccnc2)C(C)C)CC2(CCOCC2)CO1 c1(COC)cc(=NCCC2CCC(NC(c3csnc3C)=O)C2)[nH]cn1 CC(CC(F)(F)F)C(=O)NCCCOCCCNC(=O)C(O)C1CC1 N1(c2cc(C)nc(CO)n2)CCC2CCC(NC(C3(C(F)F)CCCC3)=O)C1C2 C(=O)(CCCC(F)(F)F)NCC(C)(Cn1cccn1)NC(c1occ(C)c1C)=O N1(C(c2cc(CCC)[nH]n2)=O)CC2(COC(CNC(=O)C(C(C)C)OC)C2)C1 Cc1cc(Cl)c(C(=O)NC2CCC2NC(c2ccnc(O)c2)=O)cc1N C(C(=O)N(C)CC1CCCC1)(C(C)O)NC(C(C)CO)=O CC(N=[N+]=[N-])C(=O)N1CCC(C(=O)NOC2CCCCC2OC(F)F)C1 n1(C(C)C)cc(C(=O)NCC(CO)NC(=O)C=CC2CCCO2)c(Br)n1 C(=O)(C1CCCc2nc[nH]c21)N1CC2(CC(CNC(C(C)OCCCC)=O)C2)C1 C(=O)(CS(=O)(=O)CC(=O)NC1CCCCC1NC(c1cnc[nH]1)=O)OC C=CCC(CC(=O)N(C1CSC1)C)NC(=O)CC1CCCCC1 C1(NC(Cn2ncn(C)c2=O)=O)CC2CC(C1)N(C(C1COC(=O)C1)=O)C2 O=C(CCCC1CCC1)NC1(C(=O)NC2CC(c3ccccn3)C2)CC(O)C1 NS(=O)(=O)N1CCC(C(=O)NCCNC(c2coc(C(F)(F)F)n2)=O)CC1 C(=O)(C(C(C)(C)C)N1CCNC1=O)N(CC(C)NC(CCOC(C)=O)=O)C CC1CN(C(=O)C(=O)NCCOc2cccnc2)CCC1C c1(OCC)ccc(C(=O)NC2CC2C(=O)Nc2cc(Br)cc(I)c2)c([N+](=O)[O-])c1 N1(C(Cc2cc(CC)no2)=O)CC(CNC(c2scnc2C2CC2)=O)CC(C)C1 Cc1ccc(C(=O)C(N2CCC(NC(c3nocc3C)=O)CC2)=O)cc1 c1(CCCC(=O)NCC2(CNC(C3(C(N)=O)CC3)=O)CC2)ccc(F)cc1 C1(CC)CCC(NC(c2cnc(C)cn2)=O)CC1.c1(C2=CC(=O)N2)cccnc1 CCC(CC(C)C)C(=O)N1CCC(N(C)C(c2ncncc2F)=O)C1 N1(C(C(CC)SC)=O)CCN(C(C23CC(C2)S(=O)(=O)C3)=O)C2CC12 C(=O)(C1=NN2CCCN=C2N1)NC(C)(C)CCNC(C1CCC(CO)CC1)=O c1(NC(C2(F)CN(c3cc(OC)nc(OC)n3)C2)=O)ccc(C#N)c(Cl)c1 Cc1cc2cc(C(=O)NCC3CCC(C4CCC4)CC3)ccc2cn1 C(C(CO)(CO)NC(=O)Cc1nocc1C)N(C(C(COC)NC(C)=O)=O)C C(CCCCCCC(=O)N1CC(CNC(c2ncc[nH]c2=O)=O)C(C)(C)C1)SC N1(C(C2N(C(C)=O)CSC2)=O)CC2(CCCC2NC(C2CC(=O)NC2(C)C)=O)C1 C1(C(=O)NCC(C)CNC(c2noc(C3CC3)n2)=O)CCC(N(C)C)CC1 C1(C(=O)NC(CC)C(=O)NC)CN(C(c2nccn2C)=O)CCC1(C)C c1(CC(N2CC(C)(NC(C(COCC)C)=O)C2)=O)ccc(O)c(OCC)c1 n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CN(C(=O)C(C)NC(N)=O)CC2(C)C)n1 C(=O)(CC(C)(C)COC)N1C(C)CC(NC(C2CN(C(CC)CC)C(=O)C2)=O)C1 c1(C(N2CCN(C(c3c[nH]c(=NC)s3)=O)CC2)COC)c(C)cc(Br)cc1F c1(C(=O)NC(CNC(C(CCC)C#N)=O)C2CC2)ccc(O)c2c1CCCC2 S(=O)(=O)(c1cccnc1N(C)Cc1ccc(C)s1)NC(c1cc(C)on1)C C1(NC(COCC(C)C)=O)CCCN(C(c2cc(-c3ccccc3)co2)=O)C1C C1(O)(C(=O)NC2CCN(C(=O)OC)CC2)CCN(C(C2CC23CCOC3)=O)CC1 c1(C(N(CCCCN(C(C2C(C)C2)=O)C)C)=O)c(O)nnc2c1CCCC2 C12(NCCn3ccccc3=O)C3C4C1C1C2C3C41CO.C1(C=O)C2CCC(F)(F)C12 C1(C(=O)NCCN(C(CCc2cc(C)no2)=O)C(C)C)CCC2C1C2(F)F C1(N(C)C(C2(F)CCC2)=O)CC2CC1N(C(=O)CC1C=CCC1)C2 c1(C(=O)NCC2(F)CC(NC(C3C(C)CC=CC3)=O)C2)ccc2ncsc2c1 N1(C(C2=NOC(CNC(c3scc(C)c3)=O)C2)=O)CC(C)CCC12CC2 c1(NC(CNC(C=CC(CC)=CC)=O)C)nc2c(cc1C#N)CCC2 c1(C2CC2)cccnc1Cl.Cc1cc(C(N2CCCC2CCNC(=O)C2CC2)=O)ns1 c1(OC)cccc(CCC(N2CCCC(NC(=O)C(C)(C)C(N)=O)C2C)=O)c1F c1(C(C)Nc2nccc(CC#N)n2)ccc2ccoc2c1.C1(C)CCN(CCF)CC1 C1(=O)C(C)(CSC)N1.c1(C(=O)NCCN(C)CC)cnc(=N)[nH]c1 C(CCC(=O)NCC1CNC(=O)CO1)(C(C)C)NC(C1C(C(=C)C)OCC1)=O c1(C(=O)Nc2cc(C=O)ncc2)oc(C)cc1C.C#CCN(CCOC)C1CC1 c1(NC(c2cncc(OCC)c2)=O)cc2c(cc1NC1CC1)n(C)c(=O)n2C C1(NC(=O)NC(c2ncccn2)CC)CCOC(c2cccc(F)c2)C1 c1(OC)ccc(OC)c(C(O)CNCCCC2(O)CC2)c1 N1(CC(N2CC(N(C(=O)CC3CC3C)C)C2)=O)C(=O)c2ccccc2C1=O NCS(=O)(=O)CC1CC(NC(c2nnnn2C2CCCC2)c2ccco2)C1 C1(O)(CCNC(=O)CSC(F)F)CN(C(c2cnn(Cc3cccs3)c2)=O)C1 c1(CNCc2ccc(C#N)s2)cccc(N=[N+]=[N-])c1 c1(N2C(CN(C(=O)C=CC3CCCO3)C3CC3)CCC2)ncnc2c1CCC2 CC1(C)CC(C(=O)NCc2nc(CNC(C3CC4CC4C3)=O)cs2)CNC1=O Cc1[nH]c2c(C(N3CC4(CCN(C5CCC(=O)NC5=O)C4)C3)=O)cccc2c1C c1(OC)ccnc(N2CCCC(NC(=O)CCOc3ccccc3C)C2)n1.C1CO1 C1(NC(C(C)CN(C)C)=O)(CO)CCCN(C(=O)C(C)(C)C2CC2)C1 CN1CCCC(CO)C1.C1(C(C)(C)C)CN(C)C(c2cnc[nH]2)c2nnnn21 C1(C(=O)NC(CNC(C2CC(OCC)C2)=O)CC)COCCO1 Cc1cccc2cc(C(=O)O)cnc12.c1(N2CC3(C2)NC3)nc2cc(Cl)ccc2s1 N1(C(c2c(C(C)(C)C)c[nH]c2)=O)CCOC2CN(C(C3(C)CC=CCC3)=O)CC12 N1(C(Cn2c(C)ccn2)=O)CC(OC)CC1CNC(C12CSC(C1)C2)=O c1(C(=O)NC2CCN(C(CCOC(C)C)=O)CC2CO)cc(Cl)c(N)cc1F Cc1sc(N)c(C(=O)NCC2CC(NC(=O)C(C)OCC(F)(F)F)C2)c1C C(C(=O)NCCC1CSCCN1C(c1nn(CC)nc1C)=O)(C(C)C)OCCOC N1(C(C(C(C)C)OC)=O)CC2(C=C(C(=O)Nn3ccnn3)C1)COCC2 Cc1nc(NCc2ccsc2Cl)cc(N(C)Cc2ccc(C)s2)n1 C1(C(=O)NCCC(C)N2CCCC2)CC=CCN1C(=O)C=C(C1CC1)C1CC1 C(=O)(C1=CC2(CCOCC2)C1)N1CCC(CNC(C(C)Cc2ccnn2C)=O)C1 Cc1cc(C)nc(-c2cn(CC(=O)NC(C)C(F)(F)c3ccccc3)nn2)n1 c1(COCC(=O)N(CC(N2CCC(N(C)C)C2)=O)CCC)ccccc1C C1(CC(=O)NCCOCCNC(C2(C3CCCO3)COC2)=O)CCCCC1.OC N1(C(C(CC)OCC)=O)CCC(F)(CNC(C2(c3cccs3)CCCCC2)=O)C1 Cn1nnc2cc(C(=O)NC3CCC(C)(CNC(=O)CN4CCCC4)C3)sc12 CC1(C)C2CN(C(c3cccnc3CNC(C3CCC3(F)F)=O)=O)CC12 c1(OC)cc(C(=O)NCC2C=CCN2C(C2CCCOC2)=O)ccc1C(F)F C(=O)(NNc1ncnc(Cl)c1OC)c1ccc(CC)nc1CO CCC(CC)C(C)C(=O)N(CC(=O)NCC1CCC(F)C1)C1CC1 c1(C(N2CC(C)(NC(c3c(SC)nn(C)c3)=O)C2)=O)nn(C)c(C)c1Br CN1CC=C(CC(=O)N2CCC3CCC(NC(C4CCC(O)CC4)=O)C23)CC1 C1(CNC(C=C(CC)C)=O)CCN(C(C2CC2C2(C)COC2)=O)CC1(F)F Cc1cccc(C(F)(F)C(N2CC3CC2C3NC(C2CCC(F)C2)=O)=O)c1 C1(C(=O)NCC(C(=O)NC)(C)C)CC(C)CN(C(C2(CC(C)C)CC2)=O)C1 c1(C(=O)NCC2N(C(C(C)O)=O)CC2)cccc(S(=O)(=O)N=S(C)(C)=O)c1 C(Br)(C(=O)N=S(C)(=O)c1cccc(Br)c1)=CC(c1cn(C)nc1)(C)C C1(NC(CNC(N)=O)=O)CCN(C(=O)CCNc2ccccn2)CC1CO c1(C(=O)OCC)cocc1CC.C1(N(CCN(CC(=O)N)C)C=O)CCN1C1CC1 c1(C(N(CC(C)NC(c2cc(O)cs2)=O)CC)=O)ccc(C)c2[nH]c(C)cc12 C1(NC(C(C)=C(CC)C)=O)CCCC12CN(C(=O)C(c1c(F)cccc1F)C)C2 c1(C(=O)NCC2C(NC(CC3N(C)C(=O)CC3)=O)CC2)cc(C2CC2)nc(O)c1 c1(C(=O)NC2C(O)CCN(C(c3cc(C)[nH]c3)=O)C2)cnc2cc(C)nn2c1 c1(SCC(N2C(C)(CNC(C3CCC(=O)C3)=O)CCC2)=O)ccc(C#N)cc1 c1(CC(=O)NCCC(C(C)C)NC(=O)CC(C)C2CC2)ccc(Cl)cc1F c1(NC(C2C3CN(c4nccc(C(=O)OC)n4)CC32)=O)nccc2ccn(C)c12 c1(C(c2n(CCCCCC)nnn2)NCCCC(C)(C)C)ccnc(OC)c1Cl N1(C(c2ncc(Cl)s2)C(=O)NC(c2cccs2)C2CC2)CCC(C2CCCO2)CC1 c1(C(N2CCC3CC23C(=O)NCC2(O)CCCOC2)=O)cc2ccccn2c1 c1(OC)n[nH]c(C(N2CCCC2c2ncon2)=O)c1Cl c1(C(CC)NC(C2CC(F)(F)C2)(C)C)ccc(Br)c(Cl)c1 N1(C(C(c2scc(OC)c2)(C)C)=O)CC(C(=O)O)OCC12CC2 c1(C(=O)NC)cccc(C(=O)NC2CCC2NC(=O)CC2CCCCC2O)c1 CC(C)C(CC(=O)N1CCN(C)C(CO)C1)NC(c1cc(F)ccc1F)=O N1(C(C)=O)CCC(N=c2nc3c(ncn3C)c(NCCCCCO)[nH]2)CC1 Cc1cnc(CNC(=O)C(Cc2cn[nH]c2)NC(=O)Cn2ccnc2)[nH]1 N1(C(c2c(C)nn(CCO)c2)=O)CCC2(CC1)CCN(C(C1CC1C1CC1)=O)CC2 N1(C(C(=O)NCC(C)(C)O)=O)CCC(Nc2cccc(Br)c2)CC1 c1(OCC(=O)F)cccc(OC(=O)CC2OCCCO2)c1 C1(C)(CCC(=O)OC)CCCN1C(=O)CCCc1cccc(I)c1 c1(CNC(c2cnc(-c3ccccc3)s2)=O)cccc(OCC2CCCO2)c1 C(C(COC)C(=O)NC(CC1CC1)C(=O)N1CCOCC1)OC C#CC(CNC(=O)NCc1ccc(F)c(F)c1C)CC(C)(C)C n1(CC(=O)NCC(CCOC)NC(C2C3CCOCC23)=O)ncccc1=O c1(NC(C2CCN(C(C(C(=O)OC)C)=O)CC2O)=O)c2c(nn1C)CCC2 c1(C(=O)NCC2C(C)CN(C(=O)C=CC(=O)OC(C)(C)C)C2)ccc(O)c(CO)c1 c1(C(N2CC(C)(NC(C(CCC)C)=O)C2)=O)cc2cc(N)ccc2[nH]1 C(CNC(C1C(C)CCN1C(=O)CCc1conc1C)=O)(CC(C)C)OC C1(NC(c2c(C)scc2)=O)CCC2(CC1)CN(C(=O)CCCc1ncco1)C2 C(=O)(N=c1ccc(C(O)C2CC2)n[nH]1)NCc1c(CC)non1 C1(C(N2CC(NC(C=CC(=O)N(C)C)=O)C2)=O)CCN(C2CC2)C1=O c1(C(C)=O)ccc(NC(C2(S(C)(=O)=O)CC2C(F)(F)F)=O)cc1 N1(C(C2(C(C)(C)OC)CC2)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C(CF)C1 c1(C(N2CC(C(=O)NC(C(C)C)CNC(=O)CN(C)C)C2)=O)c(F)cccc1Cl C1(C(N2CC(C)CC(NC(COCCC)=O)C2)=O)CCC2(CC1)CC(O)C2 c1(C(N(CCOCC(COCCOCC(=O)OC)O)C(C)C)C)cccc(Cl)c1 C(=O)(C1=CC2(CCOC2)C1)NC(CCOCC)C(=O)NCc1cc(CC)no1 c1(C(N2CCCC(C(C)C)C2)C(=O)NCCOC)nc(Br)ccc1F c1(OC)cc(C(N2CC(NC(=O)C=CC(C)(C)C)C(O)C2)=O)c(O)c(Cl)c1 c1(C(N2CC(NC(C(C(CC)C)O)=O)C2)=O)c(Br)sc2ccccc12 N1(c2nc(C)nc(N3CC4CCC(C3)O4)c2)C2CCC1CC(CC)C2 C1(C(=O)NCCCCO)COCCC12CN(S(=O)(=O)c1cccc(Cl)c1)C2 c1(CNC(C2(C(F)F)CCCN2)=O)sccc1Br C1(C)(NC(CC2CC(C)(C)C2)=O)CCN(C(c2ccccc2N2CCCC2)=O)C1 N1(C(C2(CC=C)CCN(C(=O)C(C)OCCCC)C2)=O)CCN(C)C2(CC2)C1 N1(C(CN(CCOC)C(C2COC(C)C2)=O)=O)CC(C)(N(C)C)C1 N1(C(CC(C)O)=O)CCC(C)C(CC(=O)NC2CC3(CCC3)C2O)C1 c1(OC)ccc2oc(C(N3CCC4CCC34CNC(=O)CC(C)(C)O)=O)cc2c1 CC1CN(C(=O)CC(CNC(C2CCC(C)(C)OC2)=O)C2CCC2)CC(=O)N1 Cc1cn2c(n1)C(C(=O)NCCCNC(C1(C)C=CCC1)=O)CCC2 c1(N2CC3CC(NC(c4cc(CCC)[nH]n4)=O)C3C2)cc(C)c(C#N)cn1 N1(C(C=C(CC)CC)=O)CCN(C(C2CCC(=O)N(CC)C2)=O)C(C2CC2)C1 c1(CNCC2N(C(C(CSC)(C)C)=O)CCCC2)cc2cccnc2[nH]1 c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)CC(C)C2)cnc2ncccc2c1 c1(C(=O)OCC(C)(O)CO)nc2nc(O)c3ccccc3n2n1.n1(C)nnnc1Br c1(NC(=O)C(N2CCN(C3CCCC3)CC2)C2CC2Cl)nc2ccccc2s1 N1(C(c2cn(C)nc2N)=O)CCN(C(=O)CCS(N)(=O)=O)C(CO)C1 Cc1cc(C(N2CC(NC(C3CC4CCC(C3)O4)=O)C(C)C2)=O)n2nccc2n1 C1(C(=O)NC(CCNC(CCc2cc(C)n(C)n2)=O)C)CCc2c(nnn2C)C1 CCCCS(=O)(=O)CC(=O)NC12CCCC(NC(c3ccns3)=O)(C1)C2 C1(F)(N(C(=O)NC(C)CCC2CCCO2)C2CC2)CCCC1 Cc1nc(C)c(C(=O)NC(C2CCCCC2)CNC(C2C(Cl)(Cl)C23CC3)=O)[nH]1 c1(NCCCC(C)NC(c2ccnn2C(C)(C)C)=O)ncc(C#N)cc1F c1(OC)ccc(NC(C2CC(O)CN2Cc2ccnc(Cl)c2Br)=O)cc1[N+](=O)[O-] CCC(O)C(C)(C)C(=O)NCC1C=CC(NC(=O)CC2CC(C)C2)C1 C12(NC(=O)Cn3ncnn3)CC3CC(C1)CC(NC(C1CC1Cl)=O)(C3)C2 C1(C(N(C2COC(C)(C)C2)C)=O)CCN(C(C2CCCC(C#N)C2)=O)CC1(C)C C1(NC(CC)=O)CN(C(c2ccc(-c3sccc3C)s2)=O)C2(CCCOC2)C1 C1(CC(=O)NCC(CSC)OC)CC(O)CN1C(=O)C=Cc1ccsc1 Cc1cc(N(C(=O)COC(=O)CC2CCCNC2)C2CC2)n(C2CCS(=O)(=O)C2)n1 C1(CNC(C=CC(CC)=CC)=O)COCCN1C(=O)Cn1cccn1 N1(C(C2CCCC(C)C2)C(=O)NCCC#N)CCCC2(CCCC2)CC1 CCC(F)(C(=O)OC)C(=O)N1CC2C(N(C)C(c3cc(F)cnc3O)=O)C2C1 Cc1cnc(C(=O)NCCCCCCNC(C2(CF)CC2)=O)c(O)c1 C(c1ccc(F)cc1)=CCC(=O)N(CC(C)NC(=O)C=Cc1ccsc1)C c1(C(N2CC=C(CNC(CCOC)=O)CC2)=O)cc2c(occcc1)=CC=2 Cc1nc(C(N2CCSCC2CCNC(=O)C(N2CCCCC2)C)=O)c(C)s1 c1(C(N2CCN(C3CN(C(c4nc(Br)c[nH]4)=O)C3)CC2)=O)ccc(O)nn1 c1(C(N2CCC(c3n(C)ncc3)C2)C(=O)NCC2CCOC2)ccc(Cl)cc1Cl C1(CNC(Cc2cn(CC)nc2)=O)CN(C(=O)CC2COC(=O)C2)CC(C)(C)C1 C1(N(C(c2csc(Cl)n2)C(=O)NCCCC)CCO)CCCN(C(=O)C2CC2)C1 N1(C(c2c(C)ccnc2)=O)CC2(C1)CN(C(C1(C)CC1Br)=O)CC2CO N1(C(=O)NN2CCSC(C)(C)C2Br)CC2(Cc3cn(C)nc3)CC1CO2 Cc1ncnc(Cl)c1C(=O)NCC1CCCN1C(=O)C1CC1 c1(NC(C2C(NCc3ncc(C)c(Br)c3)C2)=O)n[nH]c2c(Cl)cccc12 c1(C(N(C(C#C)C)C)=O)cccnc1CNC(c1coc(C)c1)=O C1(O)(CN(C(=O)CN(S(C)(=O)=O)C)C)CCCN(C(c2cc(CSC)on2)=O)C1 c1(C(N(CC(C)NC(c2c(C)cns2)=O)C)=O)nccnc1N C(c1ccoc1)=CC(=O)NCCN(CCC)C(C1CC1OCC)=O Cc1oc(CNC(=O)CC2C=NN(C)C2=O)nc1C(N1CCC(C(F)F)C1)=O N1(C(c2cccc(CC)c2)=O)CCC2(CCN(C(C)C)C2)C1 C1(C(N2CC3CN(C(C(c4ccccn4)CO)=O)CC23)=O)CN2CCC1CC2 c1(N2CC(N(C(=O)CSC(C)=N)CCC)C2)ncnc2ccc(OC)nc12 Cc1sccc1C(N1CCC(CNC(=O)C(C2CCOCC2)O)C1)=O Cc1cnc(C(=O)NCC2CC2NC(c2csc(-c3ccccc3)n2)=O)cc1Cl C(=O)(CC(C)C(F)F)NCC(=O)NCC(=O)NC1(CC)CCOCC1 c1(C(=O)NC)cc(S(=O)(=O)NC(CC)(CC)C(N)=O)ccn1 CCCC(CC(C)C)C(=O)N1CCC(CNC(=O)C(C(C)(C)C)OC)C(C)C1 C1(NC)CCN(CC2CC(O)C2(C)C)CC1 C(=O)(CCCCC(N)=O)NC(CC)CN(C(=O)C=CC(c1ccccc1)=O)C C12(C(=O)NCC(c3ccccc3)N(C(CN(C)CC)=O)C)CC(F)C1C2 O=C(N=c1ccc(-c2nn[nH]n2)n[nH]1)c1cccc(Cl)c1Cl c1(NC(c2ncccc2NC(C2CC2F)=O)=O)cc(F)ccc1Br Cc1ccccc1C(=O)NC(CNC(C1CC12CC2)=O)C1CC1 C=CCC(C)(CC)C(=O)NC1(CC(=O)NCC2(CO)CC3CC3C2)CCCCC1 C(CCC(=O)NO)NC(C1N(C(C)C)CCC1)=O.N12CCC(C1)C(C)(C)C2=O N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CNC(=O)CNS(C)(=O)=O N1(C(CNC(=O)OC)=O)CCC(OCCNC(=O)C(C)(CO)N(C)C)CC1 CC1CCCN(C(=O)Nc2cccc(I)n2)C1C(=O)O c1(C(=O)N)conc1C1CC1.CC1C(=O)NC(C)CCN1C.N(C)C Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(C3(O)CC3(C)C)=O)C(O)C2)=O)c1 c1(C(=O)NCC(C)(C(C)C)NC(c2oc(CC)c(C)c2)=O)cc2ccccn2n1 C1(NC(c2c(C)cc(CC)o2)=O)CC2CC(NC(=O)CCC3CCC(=O)N3)CC12 C(=O)(C(C)C(C)S(C)(=O)=O)N(CC(C)(F)Cn1cc(C2(O)CCOCC2)nn1)CCO c1(C(N(C(C)CNC(=O)CCCC(F)F)CC)=O)sc2ncccc2c1N C=CC(O)C(C)(C)C(=O)N1CCOC(CC(=O)NCc2cc(F)ccc2Cl)C1 C1(CC(=O)NCC(O)C2(Cl)CC2)CC2(CC2)CN1C(=O)CCOCC(F)F N1(C(C(CCC=C)NC(=O)COC2(C)CCCC2)=O)CCC2(CCCC2)CC1 C1(N(C(=O)CC2CC2)C)CN(C(c2ccccc2OCC(F)(F)F)=O)CC1F C1(OC)CN(C(=O)CNC(c2ccccn2)=O)CC1NC(=O)CC1(O)CCOC1 c1(OCC)nc(C(=O)NC(C)CNC(c2nc(O)sc2C)=O)cc2ccccc12 C1(C(N(C2CCN(C(c3ncc(C)cn3)=O)C2)CC=CC)=O)CC(C)(C)CN1C c1(C(=O)OC)[nH]c(=NCCc2cnc3n2CN(C(=O)C(F)Br)C3)nc2scnc12 Cn1nc(C(=O)NCC2CN(C(=O)C=C3CCCCC3)C3CC23)cc1C(F)F C1(C)(C(=O)NCC2C(NC(C3CC(C#C)(O)C3)=O)CCC2)CC(OC)CN1C N1(C(CCOCC#C)=O)CC(C(=O)N(C)CC2CCCC2(C)C)C(C)C1 c1(OC)cc(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(Cl)c1O N1(C(c2ccc(-c3c(C)ccnn3)s2)=O)CC(NC(C2CCCS2)=O)CC(C)C1 n1(CC(N2CCCC2Cn2ccnn2)=O)cnc2ccccc12 CC1CCCC(C(N2CCC(OCCNC(C3(c4ccccc4)CC3)=O)C2)=O)C1 C12(CNS(C)(=O)=O)CCC1CN(C(C1(Nc3cccnc3C#N)CC1)=O)C2 Cc1[nH]cc(C(=O)NCC2CCN2C(=O)C=CCF)c(=O)c1Br c1(C(=O)NCC2CCCN(C(=O)CSC(F)(F)F)C2)cccc2c1COCCN2 CC1CN(C(=O)CCc2cccc(Cl)c2)CCN1C(=O)C=CBr C12(COCCN1C)NC2.N12CCN(CC1)C2=O.c1(CC)cn(C2CC2)nn1 N1(C(C(C)CF)=O)CC(NC(c2ccc(C3CCCO3)[nH]2)=O)C(O)C1 C1(C(N(CC=C)C)=O)CCCN(C(=O)CN(CC)CC)C1 N1(C(C=CCCC(C)C)=O)CCC2(CCCN(C(=O)COCC3CCC3)C2)C1 n1(CC(N2C(CC3CC3)CC(NC(C(=O)NCC)=O)C2)=O)ccc(=O)n(C)c1=O c1(OC)cc(C(=O)NCC(O)CCNC(C2OCC2(C)C)=O)cc(Cl)c1 c1(C(N2CCn3c(C)cnc3C2)=O)ccnc2cc(Cl)ccc12 Cc1cc(C(=O)NC(C)(C)CN(C(=O)CC(C)c2ccccc2)C)nn1C N1(C(c2cc(C)sc2)=O)CCC2(CCCN2C(=O)CCC(C)C)C1 Nc1cc(F)c(F)cc1C(N1C2CCC(C2)C1CNC(=O)COC(F)(F)F)=O N1(C(=O)Cc2ccnc(O)c2)CCC2CCN(C(=O)COC3CC=CC3)C2C1 c1(C(=O)NCC(CNC(c2c(NC(C)=O)c[nH]c2C)=O)F)ccc2[nH]ccc2n1 C#Cc1ccc(C(=O)NC(CNC(c2cccc(OC)c2OC)=O)C2CC2)cn1 c1(COC)ccoc1C(N1CCCC1C1CCN(C(=O)CCC2(C)CC2)C1)=O C1(OC)CC2CC(C(=O)NCCC3(C)CCN(C(c4scnc4C)=O)CC3)CC12 Cc1ccc(C(=O)NC2CC23CCN(C(=O)Cc2ccccc2Cl)C3)cc1F N1(C(C2(CC)CC(F)(F)C2)=O)CCC(NC(=O)C(F)(F)C2CC2)CC(O)C1 C(CCC(C(=O)NCCN=S(C)(C)=O)NC(c1cc(F)ccc1O)=O)OC C(C1CCCCc2ccccc21)c1c(O)nccc1.c12nc(ccc1Cl)CN2 C#CC1(O)CCCN(C(=O)C(C2CCCN(C(=O)CSC(F)(F)F)C2)C)C1 N1(C(C(CC=C)CC)=O)CCN(C(c2csc(C(C)C)n2)=O)C2CCC12 c1(-n2cc(C(C)(C)NC(C3(C)CC3C(=O)O)=O)nn2)cccc(C(F)(F)F)c1 C(CN=c1[nH]cnc2ccc(O)cc12)(C1CCCC1)NC(C(CC)OC)=O c1(N(C(c2ccc(OCC)c(Br)c2)=O)CC)nc2ccc(C)cc2[nH]1 C(=O)(C(O)C(C)(C)C)N(CCOCCN(C(=O)C(c1ccccc1)O)C)C C1(CNC(c2ccn(C(C)(C)C)n2)=O)C2CN(C(C)C(=O)Nc3cccs3)CC12 C1(NC(c2cc(C)n(C)c2)=O)CCN(C(=O)CCc2cnn(C)n2)CC1CO N1(C(c2cnc(CC(C)C)s2)=O)CC(NC(c2cnncc2O)=O)C(O)C1 Cn1cnc(N2CCN(C(=O)CSc3ncccn3)CC(O)C2)c(Br)c1=O C1(C(N(CCN(C(=O)Cc2n[nH]c(=N)s2)C(C)C)C)=O)CCCC2(CCC2)C1 O=C(C1c2ccccc2CN1C(c1ccc(I)cc1)=O)Nc1nc(Cl)ccc1Cl C1(C(=O)NCC(CC)N(C)C)CC12CCN(C(C1CN(C)CC(C)O1)=O)CC2 c1(OC)c(C(=O)Nc2cc(C(F)F)ncn2)nc(O)nc1O.N12CCCC(C1)C2 C1(NC(=O)Cc2ccccc2F)CCCC2CN(C(=O)CCc3nc[nH]n3)CC12 c1(C(C(=O)NC(C)CC)N(CC(=O)NC)CCC)ccc(C(F)F)o1 C(=O)(C1=CCC(NC(c2csc(=N)[nH]2)=O)C1)NCC(CC(=O)OC)C N1(C(C2(CCCC)CCCC2)=O)CC2CN(C(C3CCC=CCC3)=O)CC(C1)O2 C1(OC)CN(C(C2(C)CCC(C)(C)C2)=O)CCC1NC(=O)CC1CCOC1 N1(C(c2cccc(C)c2)=O)CCCCC(CNC(=O)CC2COCCO2)C1 N1(C(C2CC(C)(O)C2)=O)CC2CC(C1)N(C(=O)CCC1CC1CC1CC1)C2 CC1CN2CCN1CC2C(=O)N(CCCNC(C12CCC(CC1)OC2)=O)C1CC1 N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(Cc3cnc(Cl)s3)CC2C1 c1(OC(CC)C(=O)NC(C)CCCCNC(=O)CC2(C)CC2)ccccc1C C1(C(=O)NCCCCCCNC(C(C)(CO)NC(C)=O)=O)CCS(=O)(=O)N1 c1(OCCC(=O)NC2(CN(C(=O)C(C)(O)C3CCC3)C)CC2)ccc(C)cc1C C#Cc1cccc(NC(=O)CN(CCC)C(C2CC3CC2CC3=O)=O)c1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NCC=CCNC(c1c(C)cncc1)=O C(=O)(NNc1cccc2c1OC(F)(F)O2)c1nc(-c2cn(C)nc2)oc1 N1(C(C2CCC(=C)CC2)=O)CC=C(CC(=O)NC2CSCC2C)CC1 c1(-n2cc(NC(N3CCC(C(F)F)(CO)C3)=O)nn2)ccc(F)cc1Cl CC(C)CC(C)(C)C(=O)NCCn1cnc(C(N2CCOCCC2C2CC2)=O)c1 c1(C(N)=O)ccc(C(=O)NC2CCCC2NC(C2CC3CC3C2)=O)cc1 N1(C(C2C(CC)OCC2)=O)CC2=C(C1)CN(C(c1ccc(F)cc1F)=O)C2 C(=O)(C1CCCc2nncn21)NCC(CC(C)C)NC(C1(C2CCC2)CC1)=O c1(C(=O)NCC(CN(C(C(C)OC2COC2)=O)C)(C)C)cnc2n1CCCCC2 O=C1NCCOCC1NC(C1C2CCC(C2)C1NC(c1cncc(O)c1)=O)=O Cc1ccc(C(=O)NC2CC(O)CN(C(c3ccc(O)cc3)=O)C2)cc1C c1(NC(c2n(CC)ncc2Br)=O)cc(Cl)cc(Br)c1I C1(NC(C(C)(C)NC(C)=O)=O)CCN(C(c2[nH]c(=N)sc2C(F)(F)F)=O)CC(O)C1 c1(C(C(=O)N)N(CCC#N)C)nc(Br)ccc1C.c1(OC)ccc(C(C)(C)CO)cc1 c1(CNC(CC2N(C(C3(SC)CCC3)=O)CC2)=O)ncccc1O C1C(C)S(=O)(=O)CC(=O)N1.C1(SC)CN(S(C)(=O)=O)C1 Cc1csc2cc(C(=O)NC3CC3CNC(=O)C(N)=O)[nH]c12 C(=O)(C(CCC(N)=O)NC(=O)CCCN(CC)CC)N1C(CC)CC(C)C1 c1(CNC(c2cccc(-c3ccncc3)c2)=O)ccc2c(c1)CCNCC2 N1(C(CN(C(CC2ON=C(C)C2)=O)C)=O)CCN(C(=O)C=CC(C)C)CC1 N1(C(COCCC=C)=O)CC2CN(C(c3cnc(OC)c(Cl)c3)=O)CC2(C)C1 C(=O)(CC(C)C(C)(C)NC(c1sc(C)cc1C)=O)NC1CC(C)(CC)C1 C=CC1(O)CC(NC(C2(Br)CCC2c2nnc(CC(=O)OCC)o2)=O)C1 Cc1ccc(C(=O)N(C2CCCC(N(C(=O)COCC(F)F)C)C2)C)nn1 c1(C(=O)NCCCN(C(=O)C(C)C2CCC2)CC)cc2ccncc2s1 N1(C(C2(C(N(C)C)=O)CC2)=O)CCCC(Cn2cc(C3CCCO3)nn2)C1 Cc1ncc(CC(=O)NC2(CNC(c3csc(-c4ncccn4)n3)=O)CC2)o1 C1(C(N2CC(N(CC(C)C)C)C2)=O)CCCN1C(=O)COCCCF Cc1noc(C2CC2)c1C(=O)NCC1(C)CCCN1C(=O)CC1(C)CCCCC1 c1(C(N2CC(NC(c3c(C)sc(CC(C)C)n3)=O)C2)=O)sccc1S(N)(=O)=O N1(C(C(CC)OC2CCCC2)=O)CCC(OC2C3CN(C(=O)CC#N)CC23)CC1 N(C(=NCc1ccc(F)cc1)N1CCC(F)C1)C(c1cc[nH]n1)COC C1(CC(=O)NC2C(NC(c3cnc(C)s3)=O)C2)NC(=O)CNC1=O N1(C(C(c2cnccn2)C)=O)CC=CC1CNC(c1n[nH]cc1C1CC1)=O c1(C(N2CCC(N(C(C3CC4CC4CC3C)=O)CC)C2)=O)ccnc2ccsc12 CC1CCCn2cc(C(N3CC(O)(CNC(=O)C(c4ccccc4)O)C3)=O)nc21 C1(C(=O)NCCCCCNC(c2cc(OC)ns2)=O)CCC2(CC1)CNC(=O)C2 CC(C)(CS(C)(=O)=O)C(=O)NC1CN(C(=O)CC2=CCCC2)C2(CCOC2)C1 C1(NC(C2N(CC)CCC2)=O)CCCCN(C(c2cc3ccccc3[nH]2)=O)CC1 CC1CCC(NC(=O)CS(C)(=O)=O)CN1C(=O)COc1ccc(Cl)nc1 Cc1ccc(-n2nnnc2N2CCC(CC(=O)NC(C)COC(C)C)C2)cc1 c1(NC(c2cc(C)c(Br)cc2)C(O)C2CC2)ccc2c(=O)[nH]ccc2c1 Cc1noc2cc(C(N3CC4CC(NC(=O)CC(C)(F)F)CC4C3)=O)ccc12 C1(CNC(C(C)(C)SCCOC)=O)CN(C(=O)COCC2CCCO2)CC1(F)F c1(C(=O)NC2C(C)N(c3cnc(F)cn3)CCC2)cnc2cnccc2c1 c1(C(=O)NC2C3OCC(NC(c4occ(C)c4)=O)(C3)C2)cccc(O)c1[N+](=O)[O-] N1(C(C(N(C(CCC(C)=O)=O)C)C2CC2)=O)CC(C)C(C2CC2)C1 N1(C(CCN(C)CC)=O)CCC(CC)(NC(c2nccnc2C)=O)CC1 c1(C(N(C)CC2(NC(C=C(CC)C)=O)CC2)=O)nccc(Cl)c1C N1(Cc2cc(OCC#C)c(OC)cc2)CC2C3C=CC(CC3)C2C1 c1(-c2cn(CC(=O)N(C)C)nn2)nnc2n1CCC2.N12CCCC1(C)OC2=O C(=O)(C1=COCCO1)N1C(CNC(c2ccc(CN3CCOCC3)o2)=O)C=CC1 C(c1ccc(=N)[nH]c1C)=CC(N1CC(C(N)=O)(CNC(CCC(C)SC)=O)C1)=O C(=O)(C1=CNC2=NCCCC2=C1)N1C(CNC(=O)CCC2CCCCCC2)CC1 C1(C(=O)NC(C)CC(N)=O)CC2CCC(C1)N2C(C1CC1(Cl)Cl)=O C(=O)(C1=CCCCC1)N1C(C(C)NC(c2csc(O)n2)=O)CCCC1 N1(C(C2CN(SCC)C(=O)C2)=O)CCC(C(=O)NC2CCNC(=O)C2)CC1(C)C c1(CNC(C(=O)NC(C2CC(C)C2)C)=O)cccc(CN)n1 C(CN=c1[nH]c(N2CCC(S(C)(=O)=O)C2)nc2c1CCCC2)OC C1(c2cn(CC(CCNC(C(CC)CCOC)=O)(F)F)nn2)CCCCN(C)C1=O C1(C)(C(=O)NCCCN(c2ccccc2)CC)CCCN(C(=O)CCN(C)C)C1 N1(C(c2[nH]c(=NC)sc2)=O)CCCCC(N(C)C(c2ncc(F)c(OC)n2)=O)C1 CC1(C)C2CCC1(C(=O)NC13CC(NC(c4cc(Cl)no4)=O)(C1)C3)CC2 CC1=C(F)CN(C2CC3CC2N(C(=O)CCCSc2ccc(Br)cc2)C3)CC1 C1(CC)CN(C(=O)CCCC(F)F)CCN1C(C1CCCN(C(C)C)C1)=O C1(C(=O)NCC(=O)OCC)CCN(C(=O)Cn2nnnc2C)C1 Cn1cnc(C(=O)CNC(C(CCCO)c2ccccc2)=O)c1 C1(C(N2C(CN(C(=O)Cn3ccc(C4CC4)n3)C)CCC2)=O)CC12CC(C)(C)C2 Cn1cccc1C(=O)NCC#CCNC(c1cnc(-c2ccccc2)o1)=O CON(CCO)C(=O)c1cc(CCNC(=O)CC(C)COC(C)C)on1 C(=O)(CC(C)C(=O)NCC1CC1CC(=O)Nc1cnn(C(C)C)c1)OC N1(C(C(C(C)NC(=O)CCCC2CCCO2)C)=O)CC2(CCC2(C)C)C1 c1(CC)cccc(C(=O)NC2(C)CN(C(C3CCOC3C(F)(F)F)=O)C2)n1 CC(C)(C)CN=C(NCC1(O)CCOC1)NCC(C)(O)C1CC1 c1(C(N2C(C)C(NC(=O)CCC3CCC3)CCC2)=O)ccnc2ccnn12 C(=O)(C(C)CC(F)(F)F)NC(CC#CC)C(=O)NC1(C)CN2CCC1CC2 CCC(C)(C)CCCC(=O)N1C(CC(=O)NC(C(C)C)C(C)C)C2CCCC12 C1(C(=O)N(CCCc2c(C)cccn2)C(C)C)CC2(CC(NC(N)=O)C2)C1 O=C(CCC(=O)c1ccc(F)cc1)NCCOCc1cn(CC2CCCO2)nn1 Nc1cc(F)c(C(=O)NC(CNC(=O)CCC2CC2)CO)cc1F c1(C(=O)NC(CCC)CCCNC(=O)C2=C(C)CCC2)cncc2ncccc12 C1(N(C(=O)C(c2cccnc2)OC)CC)CCCN(C(C2CC(F)(F)C2)=O)C1 c1(C(=O)NC2CCN(CCCCN3CCCC(O)C3)CC2)ncc(F)cc1F C(CCOCCO)(C(=O)N1CCC(C(=O)OC)O1)NC(C1(C=C)CCOCC1)=O C1(NC(CC(C=C)CC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC12CCC2 C1(CNC(COC)=O)CN(C(c2ccsc2C(F)(F)F)=O)CC1c1cncn1C c1(N2CCC(CSC)C2)nc2c(c(=NCc3nc(Br)cs3)[nH]1)SCC2 C=CCC(CNC(c1sccc1F)=O)NC(=O)C(F)n1cccn1 N1(C(c2ccc(C)cc2)=O)CCC(F)C(NC(=O)COc2ccccc2Cl)C1 N1(C(CC2(C=C)CN(C(C(C)OCCC=C)=O)C2)=O)CCC(C)CC(C)C1 CC1(C)CC(NC(=O)Cc2cn[nH]c2)CN(c2ncc(Cl)cn2)C1 c1(C(=O)NCC23CC2CN(C(=O)CCn2ccnn2)C3)cncc2nc(O)[nH]c12 n1(CC)ncc(C(=O)NC2CC(C(=O)NC3CCOCC3CC)C2)c1C C(=O)(C1=CC2CCCCCC12)N1CC2CCC(NC(C(CCC)(C)C)=O)CC2C1 C(=O)(C(C)(O)C(C)C)N(C1CCCN(C(=O)OCCc2cn(CC)nn2)C1)CC c1(C(N(C(CCNC(Cc2cn(CC)nc2)=O)C)C)=O)ccncc1CC c1(C(=O)NCC(N(C(=O)C(F)(F)c2cscn2)C)C2CC2)cccc(Cl)c1 C(=O)(C1=C(Cl)CCC1)NCCCCN(C(C1N(C(=O)NC(C)C)CCC1)=O)C N1(C(C(C)(C)C2CC2)=O)CCN(C(C2C=CCC2)=O)C(CCO)C1 c1(-c2ccc(N(C)CC3CCCN(C)C3)cc2)ccc2nccn2n1 c1(OC)ccc(CC(N2CC(NC(C3CCC(CN(C)C)O3)=O)C2)=O)nc1 Cc1ccc(OCC(=O)NCC2(C)CN(C(=O)CCCC(C)=O)CC2C)cc1C c1(CNC2CN(C(Cc3ccn(CC)n3)=O)C2)cccc(C(=O)O)c1F N1(C(C2CN(CC(C)C)C2)=O)CCCC(CN(C(=O)CCN(C)C2CC2)C)C1 c1(C2(NC(CC3CCN(C(=O)CCc4ccco4)C3)=O)CCCC2)ccc(F)cc1 CC(c1ccccc1F)=CC(=O)NC(C)(C)C(C)NC(c1c[nH]cc1Br)=O c1(C(N2CC(NC(=O)CN3CSCC3=O)C(F)C2)=O)oc2ccccc2c1Cl C12(NC(C=CC=CCC)=O)CCCC1N(C(=O)CCOCc1ccccc1)CC2 c1(C(=O)NCC(CO)NC(CCC(C)CN(C)C)=O)c[nH]c2cccc(C#N)c12 C1(C(=O)NCC(C)(F)F)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C2C(C(=O)NCc3ccc(C)s3)C2)cccc(C2=CCS(=O)(=O)CC2)c1 c1(C(=O)NC(c2ccc(C#N)cc2F)C)cn2cc(C(F)(F)F)ccc2n1 C1(C(N(C(C2CCOCC2)C)C)=O)CC(C)(C)CCN1C(C1CCC1Cl)=O c1(C(=O)NC2(CNC(c3ccc(O)nc3Cl)=O)CCC2)ccnc2ncnn12 Cn1ncnc1CNC(c1cn(CCNC(C2CCCC2)=O)cn1)=O C1(C)(CNC(CC2(CSC)CC2)=O)CCCN1C(=O)Cc1ccc(C)nc1 CCC(C)(CO)C(=O)NCc1ccoc1C(=O)Nc1cccnc1C1CC1 c1(C(CC(=O)NCC(n2cc(C(=O)OCC)nn2)C)C)ccc(F)c(F)c1 N(C(=NCCc1ccn(C(C)C)n1)N1CCC(c2ccccc2Br)C1)CC(C)CO c1(C(=O)NCC2COCCN2C(c2cc(Cl)c(Cl)[nH]2)=O)c[nH]nc1[N+](=O)[O-] c1(OC)cc(F)c(Nc2cc(OC)c(C)c(OC)c2)cc1Cl C=CCCCCC(=O)N1CC(C(=O)NCCC(C)c2cn[nH]c2)CCC1C CCCCCCn1nnnc1C1(NCCCC2CCOC2)CC(CC)C1 Cc1nc(C(=O)NCC(C)(CO)NC(c2cscc2Cl)=O)nn1-c1ccccc1 c1(OC)ccc(CC(O)C(=O)N2CCCC2C(C)NC(=O)C(C)(F)F)cc1 C(N=c1[nH]cnc2cc(F)ccc12)C1N(C(c2sc3n(C)nc(C)c3c2)=O)CC1 N1(C(COC(C)C)=O)CCCCC1C(=O)Nc1ccnc(N(C)C)c1 N1(C(c2cccc(C)c2F)=O)C2CCC1CC(C(=O)NCCCC(C)(C)C)C2 c1(C2CC2C(=O)NC2CC(NCC=Cc3ncc[nH]3)C(O)C2)ccc(CO)cc1 N1(C(c2c(C)nc(C(C)C)o2)=O)CCN(C)CC1CNC(C1CC12CC2)=O C#Cc1ccc(F)cc1C(=O)NCC1CCCC1NC(=O)CCC N1(C(CO)=O)CCCC(CN2CCN(C(C3N(CCC)CCC3)=O)CC2)C1.OC c1(CC)cc(C(N2CC3CC2C3NC(=O)CC2CC3CCC2C3)=O)c(C)o1 N1(C(C(C)NC(CC)=O)=O)CCCCC1C1(NC(=O)C=CCN2CCCC2)CC1 c1(CC(=O)NC(C(C)(C)C)CNC(c2cncc(F)n2)=O)ccc(C#N)cc1F C1(CCC(=O)NCCC2CC2)(NC(=O)CCC2CC2)CCCCC1 Cc1[nH]nc(C(=O)NCC2CCN2C(C2CC(F)(F)CCC2(C)C)=O)c1[N+](=O)[O-] CCC(CC)(CO)C(=O)N1CCCOC(CNC(c2cn(C)nc2C)=O)C1 C1(C(N2CC3(CC(OC)C3)C2)=O)CC12CCN(c1ccc(SC)cn1)CC2 CC(C)CC(CNC(=O)CCc1ccc(N)cn1)NC(c1sccc1C(F)F)=O c1(NC(=O)NC(C)CO)onc2ccccc12 N1(C(c2scc(C(N)=O)c2)=O)CCN(C(C2CC2CF)=O)C(c2ccccn2)C1 c1(CNC(C2C(C3C(C)C3)C2)=O)cccc2c1CCN(c1nnco1)C2 N1(C(C(C)S(N)(=O)=O)=O)CC(NC(C2CC3(C2)CC(F)C3)=O)CC(C)(C)C1 C1(NC(=O)COCC2CC2)CC2CN(C(c3ncc(Br)cc3O)=O)CC12 Cn1cc(Cl)cc1C(=O)NCC1CCCCC1NC(c1cnccc1Cl)=O c1(C(=O)NCC2CC(CNC(=O)CC3CCOC3)C2)cnc(O)cc1F C1(C(=O)NCC(CC=C)NC(c2coc(C(F)(F)F)c2)=O)CCC2(CCC2)C1 C1(C(=O)NOCCCC2CCCCC2)CCC2(CC2)N1C(=O)C=C1CC1 n1(CCCC)nnnc1CNC(C(=O)NC(=O)CC1CC1C1CC1)C C12(C(C(=O)N(CC(C)N(C(=O)Cn3nccn3)C)C)C)CCC(CC1)OC2 C12(C(=O)NC3C(NC(C4(OC)CCC4)=O)CCCC3)CCCN(CC1)S2(=O)=O C1(NC(C(CCNC(COC2(C)CCC2)=O)O)=O)CCc2ncnn2C1 C(C(F)(F)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(SC)C1)SC CCC(CC)C(F)C(=O)N1CCCC(F)(C(=O)NCC(n2cccn2)C)C1 C1(C2CC2)(CNC(c2n(CC=C)ccn2)=O)CCN(C(=O)C=CS(=O)(=O)CC)C1 C1(CCC)CN(CCC2CCOC2)CCO1 C(=O)(CC(C)(O)C(F)(F)F)N1C(C)CC(NC(CC2(C=C)CCC2)=O)C1 N1(C(C(C)OCC=C)=O)CC(=O)NC(=O)C1 N1(C(C=NOC)=O)CCC(C)N(C(=O)CCc2ccc(Cl)cc2F)CC1 Cc1cc(C(=O)NC2COCCC2C(=O)NC2CCC(C)(O)CC2)cnc1C C1(NC(Cc2ccc(C)c(C)c2)=O)CCC2CC1CN2C(=O)CCC(F)F N1(C(=O)Nc2cc(Br)cc(I)c2O)CCn2cnc(C(F)(F)F)c2C1 C(=O)(N=c1ccc(C)n[nH]1)NC1(OC)CCC(C)C1.C(C)(=O)OC CCCCC(C)(C)NC(C1CC(C)CN1C(=O)C(F)CC1CCOC1)=O C1(C(=O)Nc2ccc(-c3onc(C)n3)cc2)CC2(CCOCC2)CO1 c1(OCCC)ccc(CNC(=O)NCC2CCC(C(F)(F)F)O2)cc1 CCN=c1ccc(C(N2CCC(N(CCO)C(C3CC(O)C3)=O)CC2)=O)c[nH]1 N(C(=NC(C)c1nn(C)cc1Br)NC(c1ccoc1)C)CCC Cc1nn(C(C)C)cc1C(c1nnnn1C1CC1)NCC1(C(C)C)CC1 c1(C(=O)NCCN(C(=O)C(CC)n2cccn2)CCC)cnncc1C C(N=c1[nH]c(=NCCC#N)[nH]c2c(F)cccc12)C1(N(C)C)CCC(C)CC1 c1(C(N2C(CNC(=O)COC3C=CCCC3)CCCC2)=O)ccc(Br)c(O)n1 N1(C(C(=O)NCC2(OC)CCCCCC2)=O)CCC(C)CC(C)C1 n1(-c2ncc(C(C(=O)NCCC)N(CC(C)(C)OC)C)s2)c(C)ccc1C C(=O)(C1CC(=O)Nc2ncccc21)NCCN(C(=O)Cn1cccnc1=O)C C1(CC(N2C(C(C)C)CC2)=O)CN(C(=O)CCCn2cccc2)CCO1 Cc1nccnc1C(=O)NC(C)CCN(C(=O)Cc1cncs1)C C(C(C)(C)C#CC(=O)NCc1csc(C)n1)NC(C(C)=CCC)=O C(=O)(CCCC(C)(C)C#N)NC(C(=O)NC(CC)(CC)CCO)C1CCC1 CC1(C(=O)NCC#CCNC(=O)C2CC2)CC12CCN(C(c1ccno1)=O)CC2 c1(CC)c(NC(N2CCCC2C2(CO)CC2)=O)cnn1-c1ccccc1 N1(C(CCC)=O)CC(CC(=O)NC(CC)C(F)(F)F)C2(CC2)C1 c1(OC)cc(C(N2CCOC3CC23)=O)c(NC(c2cccc(O)c2F)=O)cn1 C1(C#N)(C(N2CCCCC(c3n(C(C)C)cnn3)C2)=O)CC2CCC1CC2 N#Cc1c(Br)ccc(NC2CCCCCC2O)c1F N1(C(c2ccc(-n3c(C)cc(C)n3)cc2N)=O)CCN2CCCC2C1 C1(C(NOCC=C)=O)CN(C(=O)COCC2CCC2)CC12CC2 CCCC(CC1CCCC1)C(=O)NCC(CO)NC(=O)CCOC1COC1 c1(CC(=O)N(C)C)cccc(Nc2ccc(C3CCNCC3)cc2)c1 Cc1ccoc1C(=O)NC1CC(N(C)C(C2COC(=O)O2)=O)C1 c1(C(N2C(C)(CNC(C3C(CC)OCC3)=O)CCC2)=O)cc(O)cc(O)c1 CN1C(=O)CCc2cc(C(=O)NC(C(=O)O)C(C)(C)C)ccc21 C1(O)(CC(=O)NC2(CCN)CCC2)CCCCC1.CC(C)N(C(C1CC1)=O)C Cc1csc(=O)n1CCC(=O)NCCN1CCN(C(=O)CCCC2CC2)CC1 c1(C2CC(OC(C(C)C3CCC3)=O)C2)cccc(Br)c1 N1(C(CC2N(CC)CCC2)=O)CCC(NC(=O)Cc2ccc(C)s2)C1C C(=O)(C(C)C(C)c1ccccc1Cl)NCCCN(C(c1c(CC)noc1)=O)C c1(COC)nc(=NCC2(CCNC(c3cnsc3C)=O)CC2)s[nH]1 C1(NC(c2c(C)nc(CO)o2)=O)Cc2ccccc2C1NC(=O)CC1C=CCC1 N1(C(CN(C(C(C)O)=O)C)=O)CCC(CNC(C2CC2c2ccsc2)=O)CC1 c1(N2CCC(CC)OCC2)ccc(S(=O)(=O)N2CCSC2)cn1 C(C)(C(=O)NCC(O)OCC)N1CC1=O.CCCS.C1(S)CC1CC(C)C C(=O)(CC(C)CC(C)(C)C)NCC(C)(C)NC(c1cc(C#C)c(C)cc1)=O C1(CC=C)(NC(CC2C(C(=O)NCC3CC(CCC)C3)CC2)=O)CCOC1 c1(C(N2C(C)CC(O)C2)=O)ccc2c(c1)CN(C(c1ncc(Cl)cc1F)=O)C2 c1(OCCC(=O)N(CCNC(C(F)=CCC)=O)C)ccc(C)cc1C C1(C(N2CCC(NC(C3CCN(CCOC)CC3)=O)C2)=O)CCCCCC1(F)F C1(C)(C(=O)NCC2(NC(c3c(SC)ccs3)=O)CCOC2)CCC(=O)N(C)C1 C(=O)(CCS(=O)(=O)Cc1ccccn1)NCCN(C)C(C12CCCN1CCC2)=O C1(NC(C)(C)C=CC)COC(C)(C)CN1CC.C(=O)(CCCC#N)O CC(C)C(N=c1ccc2nnnn2[nH]1)C(C)NC(c1cc(Cl)cc(Cl)n1)=O c1(CNC(c2coc(C(F)F)n2)=O)n[nH]c2c1CN(C(c1cnc[nH]1)=O)CC2 CCCCCC(C)(CC)C(=O)N1C2CCC1CC(CNC(=O)C#CC1CCC1)C2 c1(C(=O)NC(C)CNC(C2CC2C2CC2)=O)cc2ccccc2n1C C1(F)(CNC(c2cnc(C)n2C)=O)CCC(CNC(=O)CCCC2CC2)CC1 c1(C(=O)NCC2CN(C(CC=C)=O)C(C)CC2)nn2cccnc2c1Br c1(C(N(CCNC(C(c2ccnn2C)OC)=O)C)=O)ncoc1-c1cnn(C)c1 C(CC(=O)NCc1nccn1C1CC1)(C(F)F)NC(c1c(CC=C)cccc1)=O c1(OC)ccc2cc(C(N3CC4CC(NC(=O)C(F)C(C)C)C3C4)=O)n(C)c2c1 N1(C(CSc2nc(C)cc(C)n2)=O)CCC2CCN(C(c3cc[nH]n3)=O)C2C1 C=CC1OCCC1C(=O)NC(C1(O)CN(C(=O)CC2(C(F)(F)F)CC2)C1)C N1(C(C)=O)CCCCC1N(C(=O)C1=C(Cl)CC1)Cc1cc(C2CCCO2)n(C)n1 C1(c2cn(CCN(C)C)nn2)CCN(C(c2ccc(F)c(F)c2)=O)C1(C)C c1(CN2CCC(O)(C(=O)Nc3cccnc3Cl)C2)ccc(Cl)c(I)c1 C1(C(=O)NCC2CN(C(=O)Cn3cnccc3=O)CC2O)COC2(CCC2)C1 Cc1nn(C2CCCN(Cc3nnc(C4CCCS4(=O)=O)o3)C2)c(C)c1Cl C12(C(=O)NC(CNC(c3ccc(CC)[nH]3)=O)C)CCC(C1)OC2 c1(C(N2C(CNC(C(CC=C)C)=O)C(C)CCC2)=O)nccc2ncccc12 CC1C(C(=O)NCC2CN(C(=O)CCSCc3ccccc3)C2)C(O)C(=O)N1C C#CCC(CC#C)C(=O)N1CC(NC(=O)CCCCCNC(N)=O)C(SC)C1 Cc1cccc(N)c1C(=O)NCC#CCNC(=O)C(C(C)C)c1ccccc1 Cc1ccc(NC(=O)C(c2ccnn2C)NC(C2CC=CCO2)=O)c(F)c1F N1(C(c2c(CC)noc2)=O)CC2(CC(NC(=O)C(N3CCCC(C)C3)=O)CO2)C1 Cc1[nH]c2ccccc2c1C(=O)NC1CCCC1C(=O)NC(C1CCOC1)C c1(N2CC(CC)C(N(C)C)C2)[nH]c(=NC2CC(CF)C2)nc2c1cnn2C(C)C N1(C(c2c(=N)[nH]cnc2)=O)CCCC1C1CCCCN1C(=O)CCSC(F)(F)F C(=O)(C(F)C(F)(F)F)N(CC)CC1CCCN(C(c2ccoc2)=O)C1 N1(C(C2(C#C)CC(=O)C2)=O)CCC=C(C(=O)NC(c2nccc(O)n2)C)C1 c1(C(CNC(c2cc(C)[nH]n2)=O)NC(=O)C(C)(O)C2CC2)ccc(F)cc1 C1(C(N2CCC(C(N)=O)C2)=O)(OC)CCN(C(=O)C=C(C)C(C)(C)C)CC1 C1(CNC(=O)CNC(=O)Cn2cncn2)CCCN1C(c1cccnn1)=O CCCCCC(=O)N1CCOC(CC(N2CCCC2CNC(N)=O)=O)C1 C1(CNC(c2ccc(C)s2)=O)CN(C)CCN1C(c1ccc(C(C)(F)F)cn1)=O c1(C(=O)NC2CC(N(C(=O)CSC(F)(F)F)C)C2)cccn2ccnc12 C1(C(=O)NC(CNC(c2c(CC)n(C)nn2)=O)C2CC2)C2CCCCCC12 N1(C(C(COC)COC)=O)CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)CCC(O)C1 C1(NC(CC=CCC)=O)CC2C(NC(=O)CCC(=O)c3cccs3)C2C1 c1(CCC)ccc(CNC(c2cc(C)[nH]n2)c2nnnn2C(C)CC)cc1 NS(=O)(=O)c1ccc(C(=O)NC(CCCCNc2nnco2)c2ccccc2)[nH]1 C1(NC(=O)CCc2cnco2)CCN(C(=O)CC2CC2)C(c2ccccc2)C1 C1(CNC(c2ccco2)=O)CCC2CCC1N2C(C1(c2ncon2)CC1)=O C12(C(N(CCCNC(=O)Cc3cc[nH]n3)CCO)=O)CCC(F)(CC1)CC2 N1(C(c2cn(C)nc2)=O)CCC(NC(c2ccc(C#N)o2)=O)C(C(N)=O)C1 Cc1cc(C(N2CC(N3CCN(C(=O)Cn4cnnc4O)CC3)C2)=O)c(O)nn1 CC(CC(=O)NCC(C)CN(C)C(C1CC(C)(C)C1)=O)c1ccco1 N1(C(Cc2c(C)nc[nH]2)=O)CCC2CN(C(=O)C(O)CC[S+](C)C)CC2C1 C1(CC=C)(NC(=O)CC2(C)CC(F)(F)C2)CCCN(C(C2CCC(C)O2)=O)C1 CN1CCN(CC(=O)NCC23CC2CN(C(=O)COc2ccccc2)C3)CC1 c1(NC(CC)(CNC(=O)C(C)Cc2ccncc2)CC)ccc(C#N)c(C)n1 c1(CNc2cc(NC(C3CC(O)CN3SC)=O)cc(F)c2)c[nH]c2ccc(F)cc12 C1(NC(C2N(C)CCCCC2)=O)CCCCCCC1NC(=O)CCc1cnoc1 CS(C)(=O)=NCC(=O)NC1CCN(C(c2ncsc2C(F)(F)F)=O)CC1CO c1(OC)ccc(C(N2CCN(C(=O)Cn3cnnc3O)C3CC23)=O)cc1Cl C(CCCC(C)NC(=O)C(Cc1ccco1)CC1CC1)NC(CCCSC)=O Cn1nc(C(=O)NC2CCC2CNC(c2cc(O)cc(=O)o2)=O)c2ccccc12 CC1CC(NC(=O)C(=O)Cc2ccccc2)CCN1C(=O)Cc1cocn1 CCC(CC)C(=O)N(C(CC)CC(=O)NCCC1(COC)CCC1)C c1(C(=O)NCC(CC)NC(c2cc(Cl)n(C)n2)=O)c(C)oc(C)c1Br c1(C(=O)NCc2c(C(=O)NC(C(C)C)(C)C)nco2)ccccc1Cl C(=O)(CCCN(C(=O)CCOC(C)CC(C)C)C)NC(C(=O)NC)C C(CCCNC(=O)CCC1CCCOC1)(c1ccccc1)NC(C=C(C)Cl)=O CCCC(C(=O)N1CC(N(C(=O)CN(C)C)CC)C1)S(N)(=O)=O c1(C(=O)NCCN2CCN(C(C3C(=C)C3)=O)CC2)ccc2ncsc2c1 C1(C(N2C(C(C)C)CCC2)=O)CCN(C(=O)COC2CC=CC2)O1 C1(CC)(NC(=O)C(C)CC(C)C)CCN(C(c2ccncc2)=O)CC1 c1(CC)sc(C(=O)NCC2CCN(C(=O)C(O)C3CCC3)C2)cc1C c1(N(CC=C)C)ccc(Br)c(S(=O)(=O)NCCc2c(F)cncc2F)n1 c1(C(C(=O)NC(c2ccc(Cl)s2)C)O)ccccn1 C1(CNC(C2(OC)CCCCC2)=O)CC2CCC(C1)N2C(=O)C(C)C1CC1 N1(C(Cc2c(OC)c(F)ccc2)=O)CC2CCCC(C1)N2C(=O)C(=O)NC1CC1 Cc1cccc2[nH]c(C(N3CCC4CCC(C3)N4C(=O)CNC(N)=O)=O)cc12 C1(C)(NC(c2ncn(CC)c2)=O)CCN(C(c2cc(-c3csc(C)n3)c[nH]2)=O)C1 C(CN=c1nc(C#N)cc(C)[nH]1)C1N(C(C(Cn2ccc(C)n2)C)=O)CCCC1 C12(NC(c3nn(CC)c(C)c3)=O)CCCC1CN(C(c1cc(C)oc1C)=O)C2 C(=O)(C(C)(C)CC(C)C)N1C(CNC(c2cnc(CC(C)C)[nH]2)=O)CCC1 C1(C(N(CC(C)NC(C2CC23CCOC3)=O)C)=O)COCCN1CC(F)F Cc1cc(Br)c(Cl)cc1NC(=O)C(c1ncccc1F)(F)F C1(C)(NC(C(C)CCN(C)C)=O)CCCN(C(=O)CC2CCC(C)C(C)C2)C1 C1(CNC(C(COC)C)=O)CC2CCCCC2N1C(=O)CCn1cccnc1=O N1(C(CC(C)OC)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C(C)C)=O)C(C)C1 c1(C(=O)NC2CC3CN(C(C4N=C(C)SC4)=O)C2C3)c(C)[nH]c2ccccc12 Cc1ccc(C(=O)NC(C2CCN(C(=O)CC3COCCO3)CC2)C(C)C)c(C)c1 c1(OC)ccc(C(=O)NCCNC(C2C3CC3C3CC23)=O)c(OC)c1Cl C(=O)(C#CC1CCCCO1)NCCCN(C(c1c(Br)ccc(C)n1)=O)C1CC1 Cc1cccc2oc(N3CCCC(CNC(=O)C(C)C4CC4)CC3)nc12 c1(C(C)C(=O)NCC2(F)CN(C(=O)CCN3CCCC3)C2)nc(F)ccc1Cl N1(C(C(C(CC)O)C)=O)CCc2cc(CNC(c3ccc(F)cc3)=O)ccc2C1 N1(C(CCC)=O)C2CCC1CC(CNC(c1ccc(OC(F)F)cc1)=O)C2 c1(C(=O)NCC2CC(NC(C(C)N(CC(F)(F)F)C)=O)C2)ccc(N)cc1Cl C(=O)(C(CC1CCCC1)CC)N1CCC(CNC(CC2(C=C)CCC2)=O)C1 C1(CNC(C2CCC(=O)NC2)=O)CC2(CCN(C(c3cc(Cl)cnn3)=O)C2)CO1 CN1CC(C)(C)CC1C(N1CCCC1(C)c1cn(-c2c(F)cccc2Cl)nn1)=O Cc1cc(C(N2CCCCC(NC(c3ccc(Cl)nc3O)=O)C2)=O)nc(C)c1 C(=O)(C1=NOCC1)N(CC(CC)NC(=O)Cc1cccc(OC(F)F)n1)CC N1(C(CC2C(C)=NN(C)C2=O)=O)CCC2CCN(C(c3nnn(C)n3)=O)C2C1 CN1N=CC(CC(=O)NCC2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1=O CCC(C#N)C(=O)NC1(C)CC(NC(c2cc(CCCO)on2)=O)C1 c1(NC(CSCCNC(CC(C)n2ccnc2)=O)=O)ccc(C2CC2)c(F)c1 c1(OCC(=O)OCC2CC(C(F)(F)F)(OC)C2)ccc(C)c(Br)c1 C1(C(=O)NCC2(C(=O)NCCSC(F)F)CCCO2)CC2(CC2)CO1 C(=O)(C1=CCc2ccccc21)NCC1C(NC(c2cc(C3C(C)C3)on2)=O)CCC1 c1(C(N(C(C)C(N2CC3(C2)CC3(F)F)=O)C2CC2)=O)c[nH]c2ccccc12 Cc1nn(C2CC2)cc1C(=O)NC1CC(NC(C2(C(=O)NCCO)CC2)=O)C1.CO c1(C(=O)NCC(CNC(C2N(C(C)=O)CC(O)C2)=O)C)cncc(Cl)c1C N1(C(C(COC)(C)O)=O)CCN(C)C(CNC(=O)Cn2nc(C)cc2C)C1 c1(NC(C2C(C(=O)OC)C2)=O)cc(C(=O)NCCCC(F)(F)F)cnc1Cl C#CC1(C(N2CCC(O)(CC)C2)=O)CN(C(=O)CCCC2CCCO2)C1 N1(C(C(C)OCCOC)=O)CCC2CCCC12C(=O)NCC1CCC(C)(CO)O1 C(=O)(CCCCCCC(=O)NC(CO)C(C)NC(=O)C(=O)N(C)C)OC N1(C(C2CC(O)C(F)C2)=O)CC2(CC2)CC1CC(=O)NC1CCOC1 C(=O)(CC1=NN(C)C(=O)C1)N1CC(CC)C(NC(c2cc(Cl)c(Cl)[nH]2)=O)CC1 CN1CC2CC1CN(C(C1CCCC(CNC(=O)CSC(F)(F)F)CC1)=O)C2 C1(NC(C2(C)COCCO2)=O)CC12CCN(C(=O)CS(N)(=O)=O)CC2 C1(CNC(c2c(CNC(CCC#C)=O)ocn2)=O)CCC(=O)NC1C C1(CNC(C(C)SC)=O)CC2(CCN(C(c3c(N)cc(C)cc3F)=O)CC2)CO1 c1(C(C)C)ncc(Br)c(=NC(CNC(C2CCC(=O)N2C(C)C)=O)CO)[nH]1 C1(C)(CNC(c2cc(C(C)C)[nH]n2)=O)COCCN(C(=O)C(C)C2(O)CCC2)C1 c1(CCNC(C(C)NC(=O)NC2CN(C(=O)C(O)CF)C2)=O)ccc(F)cc1F N1(C(C(C2CC2)OCC)=O)CCCN(C(c2n[nH]cc2C(C)C)=O)CC1 N1(C(Cc2ccc(C)o2)=O)CC(C(=O)NC2CCOCC2C)CCC1(C)C C(C1CCCC1)=CC(=O)NC1CC1NC(=O)COc1cccnc1 N1(C(C(CN(C)C)O)=O)CC(NC(C2(C)CC2)=O)C(C2CC2)C1 CCC(C)(C(=O)NCc1ccoc1C(=O)NCCC1CC(C)=NO1)OC N#Cc1cnn2cc(-c3nc(CC4CCCS(=O)(=O)C4)no3)cnc12 C(=O)(CCCCC(C)C)N1CCCC(C(C(=O)NC(C2CCCC2)CC)C)C1 C(C(CNC(=O)CC12CCC(CC1)C2)S(C)(=O)=O)NC(C(C=C)OC)=O c1(C(N2CC3CCN(C(C(C)C4CC4)=O)CC32)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 CCC(C)(C)C(O)C(=O)NC(Cc1ccco1)C(N1CCOC(CC(C)C)C1)=O C#Cc1ccnc(C(=O)NC(CCC)C(=O)N2CCOC(C3CCC3)C2)c1 c1(NCC(=O)NC)[nH]c(=NC(C)c2cnn(CC(F)(F)F)c2)nc2c1cnn2C c1(C(=O)NC(CCC)CCCNC(=O)CC(CC)C2CC2)cn2cccnc2n1 Cc1noc(C)c1CC(=O)N(C)CCC1CCCCN1C(C1CC1C(C)(F)F)=O C1(C2CCC2)(C(=O)NC2C(CNC(=O)Cc3cccc(Cl)c3)C2)CC1(F)F C1(NC(Cc2cc(C)on2)=O)CCCC2CN(C(=O)C(F)CC3CCOC3)CC12 C#CCC(CC(=O)NC(c1nnnn1C)C)NC(C1(C)CCOCC1)=O C(=O)(C1CCc2nccn21)N(C)CC1CCCN(C(c2ccc(O)nc2)=O)C1 C(=O)(C(CC(C)C)N(C)C(C(C)CC1=CCCC1)=O)NC(CC(C)C)C c1(-n2ncc(C)c2)cc(Nc2ccc(Cl)cn2)nc(C)n1.C12CCN(CC1)C2=O N1(C(CN(C(C)C)C)=O)CCCCC1C1CCCN1C(=O)Cc1ccccc1F C1(C(N2C(CCNC(C(CC)(C)O)=O)CCCC2)=O)CCCC2(CC1)CC2 C1(O)(C(C)NC(=O)CC2(C)CC2)CN(C(=O)CCCc2ccccc2)C1 C12(C)CCC(C1)N(C)C2.C(=O)(CCOCC(=O)NC1CCC1)OC c1(C(N2CCC(CC(C)C(=O)O)CC2)=O)ccc(S(=O)(=O)C2CC2)cc1F c1(OC)c(Br)ccc(F)c1S(=O)(=O)NC(c1ncccc1Br)C C(C(CC(=O)NC1Cc2ccccc2C1NC(=O)C1=CCC1)C(F)(F)F)N(C)C C(=O)(C(C)CC(F)(F)F)NC1C(CCC)CN(C(C2C=CC=CC=C2)=O)C1 c1(C(N(C2CCN(C(C34CCC3C4)=O)C2)C)=O)cccc(C#N)c1 c1(C(N2CC(CC=C)(NC(c3nc(C)sc3C)=O)C2)=O)cc(C#N)ccc1O C(=O)(CCC(O)C(C)(C)C)NCC(C)N(C(c1cc(SC)ncc1)=O)C N(C(=NCCCF)NCC(C(=O)OC(C)(C)C)C1CC1)C(CC)CC C1(F)(CNC(c2c(C)cnn2C)=O)CC2CCC(C1)N2C(C1CCC(C)(C)C1)=O CC1CN(C(c2cccc(C#N)c2)=O)CCC1N(C(=O)C1=CCOCC1)C c1(C(N(C)CC2CN(C(=O)C=Cc3cncnc3O)C2)=O)cc2ncccc2s1 c12cc(Cl)ccc1CNC(=O)N2.C1(CCS)CCCC1(F)F.C1(N)CCCC1 c1(C(=O)NCC2CCC(C)N(C(c3cc(Cl)n[nH]3)=O)C2)cccc2c1OCCN2 c1(OC)ccc(CN2CC3CC2CN3C(=O)CCNC(N)=O)cc1F C1(NC(CCC(=O)NC)=O)CC2CC1N(C(=O)CCCN1C(=O)CN(C)C1=O)C2 N1(C(c2c(C(C)C)scn2)=O)CCN(C(c2cc(CN(C)C)no2)=O)CC1CF CCCCC(C(=O)N1CC(C(N2CC(OC)CC(C)C2)=O)CC12CCC2)C(C)C C(CC1CC1)(CC(=O)N1CC2C(N(C)C)C2C1)NC(CSCC#C)=O N1(C(C2C(C)CCC2)=O)CCC(CO)(CNC(=O)COC(F)F)C1 CCC(CCC(=O)N(C(C)CN(C)C(c1ccc(C(=O)OC)s1)=O)C)OC C(=O)(C1=CC2CCCC12)NCC1CCN(C(C(C(C)(C)C)NC(N)=O)=O)CC1 C1(CCNC(c2ccn(C)c2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C1 C12(CNC(C3CC(C#N)C3)=O)CCC(NC(=O)Cc3cccc(Cl)c3)(CC1)CO2 CC1=C(C(=O)OC(c2ccc(Oc3ccc(F)c(Cl)c3)cc2)C)CCO1 N#CC1CN(C(c2cc(Cl)ncc2F)=O)CC1Nc1ncnc2sccc12 N1(C(C2(S(C)(=O)=O)CC2)=O)CC2CCCC2(CNC(=O)Cc2cccnc2)C1 c1(NCc2c(CN(C(CN(C)CC)=O)C)cccc2)ncc2ncnc-2[nH]1 CC1CN(C(c2cnnn2C)=O)CC1NC(C1(C)C=CCC1)=O N1(C(C2N(C(c3c(CC)nn(C)c3)=O)CC(C)C2)=O)CC2CC2C2CC12 C1(N(C)C)CCCC(CC(=O)NCC(O)CNC(C2CCSCC2)=O)C1 C1(C(=O)NCC2CC(F)(CNC(Cc3n[nH]c(=N)s3)=O)C2)CCCN1C=O CC1COCC(CC(=O)NCc2ccc(C(=O)NC(C3CCCCC3)C)cn2)O1 N1(C(c2n(C)cnn2)=O)CC2CCCC(C1)N2C(C12CCC(C)(CO1)C2)=O c1(OC)cncc(C(=O)NCC2(F)CCC(CNC(C3(CCF)CCC3)=O)C2)c1 c1(C(=O)NCCC2(O)CCN(C(=O)CCC3CC3(F)F)C2)cc(Cl)cnc1O c1(C(N2CCC(N(C(=O)C3=NOCC3)CCC)CC2)=O)cn2c(n1)CCC(C)C2 C1(NC(C#C)CC(C)C)CCOC2(CCC2)C1 C(C(C(=O)NC1(CO)CC(F)C1)C(C)(C)C)NC(CCCC#C)=O CC(C)CC(C)(CNC(=O)C(C)(C)O)NC(=O)CCCCc1cnn[nH]1 C#Cc1ccc(C(=O)NC(C)C=CC(=O)NCCSC(F)F)cc1 Cc1cnn(C)c1C(N1CC(NC(c2nccc(OC(F)F)n2)=O)C(O)C1)=O C(=O)(C1c2c[nH]nc2CN1C(C1CCN1C)=O)NCc1cc(OC)ncn1 N1(C(c2ccc(OC)o2)=O)CCC(NC(C2CCCS2)=O)C(O)C1 c1(-c2cn(CC(=O)NCC3CCC(CO)CC3)nn2)cc(F)ccc1CO C1(C(=O)NCC2(CNC(c3c(C)cc(Br)o3)=O)CCC2)CCC2CCC(=O)N12 O=C1NCC2(CCCN(CCCc3cc(F)cc(F)c3)CC2)N1 CC1(F)CCN(C(C2CCN(C(=O)CCc3nncs3)CCO2)=O)CC1 Cn1ccc(C(N2C3CCC(C3)C2CNC(C2CC2c2cccs2)=O)=O)cc1=O Cc1ccn(C2CN(C(=O)NCC3(C(c4ccccc4)O)CCCC3)C2)n1 C1(CC(=O)N(C2CCCC2)CCCNC(c2c(C)n[nH]c2)=O)CC(C)(C)CO1 C1(O)(C(C)C)CCN(C(=O)CC2CCCN2C(=O)Cc2ccn(C)c2)C1 Cc1n[nH]c(=NC(C)CNC(=O)COc2cnn(C)c2)o1 C(=O)(CCC(=O)c1ccc(F)cc1)NC1C(CNC(C(C)(F)F)=O)CCC1 C1(CC)C(NC(=O)CCN2CCCC2)CCCN1C(c1ccc(F)c(F)c1)=O C1(C(=O)OCc2cc(CC(CC)O)on2)N(C(=O)OC(C)(C)C)CC1(C)C c1(C(N2CCCC(CN(C=O)C3CC3)C2)=O)c(Cl)cc(Cl)c(Cl)c1F N1(C(CCNC(=O)NC)=O)CC2CC1(CNC(C1C(C(F)F)C1(C)C)=O)C2 n1(CC)cc(CC(=O)NC2(CNC(=O)C(C)C(C)(F)F)CC2)c2ccccc12 c1(OCC)ncc(Br)cc1NC(C1(C(=O)OC(C)(C)C)CC1C)=O C1(C)(NC(C2(CC#C)CCCO2)=O)CCN(C(=O)C#CC2CC2)CC1 N1(C(Cc2c(S(C)=O)cccc2)=O)CCC(C2CCCN(c3nnns3)C2)CC1 N1(C(CCn2c(C)cc(C)c2)=O)CCCC(c2ccccc2)CC1.C(C(F)F)(C(C)(C)C)N c1(OC)c[nH]c(C(=O)OC)cc1=O.C1CCCCCNC(=O)C1c1cncn1C Cc1cccc(C(=O)NCCC(C)CCNC(=O)C(F)n2ccnc2)c1C C1(C(=O)NCC#CC#CCO)(NC(c2scc(OC)c2)=O)CC(CO)C1 C1(NC(C(C)Oc2cccnc2)=O)CC(N=c2nn[nH]n2-c2cccs2)C1 C1(NC(C(CC)NC(N)=O)=O)CCN(C(=O)C(Cl)=CCl)CCC1(F)F C1(O)(CNC(C2(OC)CC2)=O)CCCN(C(=O)CCCc2nncn2C)C1 C12(c3ncn(C)c3)CC(CN1C(=O)Nc1cccc(NC(F)Cl)c1)C2 c1(CC(C(=O)OCC)NC(C)C(=O)OC)ccc2c(c1)OCCO2 CN1CCCC1C(=O)NC1CCC1NC(C1(n2ccnn2)CC1)=O N1(C(CC(C)(C)C)=O)CCOC2(CCCCC2NC(C2CCCCC2C)=O)C1 C1(NC(CCCN(C)C)=O)CC2CC1CN2C(c1ccc(C2CC2)s1)=O c1(C2C(CSCc3nc(CC)on3)C2)ccc(Br)cc1 C1(CC(=O)O)(CN2CCN(C(C(COC)NC(C)=O)=O)CC2)CC2CCC1CC2 c1(C(=O)NCC2N(C(CCCc3nnc(C)n3C)=O)CCC2)cccc(O)c1C CCCC(C)CN=c1ccc(S(=O)(=O)NCCC(O)CN(C)C)c[nH]1 c1(C(=O)NCC(CC)NC(=O)CCC=CBr)cc(N)cc([N+](=O)[O-])c1 CCC(CCC(=O)NCC1(CO)CCN(C(=O)CCCn2ccnc2)C1)OC c1(C(=O)NC2C(NC(c3c[nH]c(C)c(Br)c3=O)=O)CC2)cccn2c(O)nnc12 C1(CC)CN(C(=O)C(CO)NC(c2cc(CO)c(C)o2)=O)CCN1C C1(NC(=O)OC(C)(C)C)CCCCC1CNC(C1CN(C(=O)C(N)=O)CCO1)=O N1(C(c2cncc(C)c2Cl)=O)CC2(C1)CN(C(C1(C)CC1F)=O)CCO2 C(=O)(C(CCCC)C(C)C)NCC(C(=O)N(C)CC1CCCC1O)CC1CCCC1 N1(C(C2(N(C(=O)C=C3CCCCC3)C)CC2)=O)CCOC2(CCC2)CC1 C(=O)(C(C)(C)CF)N(C(CC)C(=O)NC1CCCC1CSC)C c1(C(N2CCC(NC(=O)CCC(F)F)CC2C2CC2)=O)ccc(Cl)c(F)c1F CCC(CN=c1ccc(S(=O)(=O)NCC2CCCS(=O)(=O)C2)c[nH]1)n1cccn1 N1(C(=O)NCCn2nnc(C)n2)CCC(C(=O)O)C1(C)C C1(C(N2C(C)CC(NC(=O)C(c3ccccn3)O)CC2)=O)CC2C=CC1C21CC1 CC1CSCCCN1C(C1CC(C)N1C(=O)CC1OCCO1)=O C1(C(=O)NCCn2cc(C(N3CC(OCC)C3)=O)nn2)CCCCS1 N1(C(c2c(CC)nn[nH]2)=O)CCC(F)(F)C(CNC(c2sc(F)cc2C)=O)C1 C1(NC(c2ccc(CC)[nH]2)=O)CCN(C(=O)C(C)CSC)C1C N1(C(C)=O)CCCc2cccc(N3CCCC3)c21.Cc1cc(C(=O)C)c(C)[nH]1 N1(C(COC2CC(Cn3cc(C(=O)OC)nn3)C2)=O)CCOC(C)C1C(=O)OC CC(C)CC(C)CC(=O)N1CCC(C(N2CCCC2CN=[N+]=[N-])=O)C1(C)C c1(C(N2CC(CCC)C(NC(c3cc(F)c[nH]3)=O)C2)=O)cccc(C)c1O N1(CC)N=C(C(=O)N2C(CN(C(c3cc(C4CCC4)[nH]n3)=O)CC)CC2)CCC1=O N1(C(C2(CC)CC(C)(C)C2)=O)CC(CNC(=O)CC2CCSC2)CC(C)C1 C1(C(=O)NCC2N(C(c3cc(CC)n(C)n3)=O)CCC2)CN(C)C(=O)CCO1 CC1C(NC(C2CCCS2(=O)=O)=O)C(C)CCN1C(=O)CC1CN2CCN1CC2 CCCC(CCCNC(c1ccn(CC)c1C)=O)NC(C1CC2(C1)CC(O)C2)=O c12ccccc1NC2=O.C1(C2CC2)(CCOCC(=O)NCC)CCCC1.C(CCF)O c1(C(=O)NCC2CN(C(c3scc(C)c3)=O)C3C2C3)ccc2nnn(O)c2c1 C1(CC(C)C)(C(=O)NC2CCC(CNC(C3(C#N)CC3)=O)C2)CCNC1=O c1(C(C(=O)NC(CN(C(=O)CC2CC(SC)C2)CC)C)(C)C)ccccc1C c1(C(=O)NC2CC(CCNC(C(C)NC(=O)OC)=O)C2)cnc(C(C)C)nc1O N1(C(C2(C=C)CCN(C(=O)CCOC3CCC3)C2)=O)CC(C)OCCC1C N1(C(c2nc(C)sc2)=O)CC2CC(C1)C2C(=O)CC1CCCC1C c1(C(C)C)ccc(C(=O)NCC2CC(F)(F)CN2C(c2cnsn2)=O)cc1F C1(C)(CNC(C(C(C)C)NC(=O)Cn2cc(CO)nn2)=O)CC2CCC1C2 C(=O)(C(C(C)NC(c1ncccc1Cl)=O)C(C)C)Nc1c(OC)cc(F)cc1 C12(CNC(c3ncn(C)c3)=O)CC1CN(C(=O)CCCC1CCOCC1)C2 C1(c2n(CCc3ccccc3)nc(-c3cncs3)n2)CN2CCC1CC2 C(=O)(CCCC(C)(C)C)N.CC1CCCc2n[nH]cc21 c1(C(=O)NC(C2(CN(C)CC)CCCC2)=O)oc(C2CC2)nc1C.N1CC(O)(CC)C1 C=C(C)c1ccccc1NC(C1CCN(C(=O)C(=O)N(CC)CC)C1CC)=O c1(CC)nc(N2CC3CC2(CNC(=O)CC(C)(C)CCOC)C3)c(F)c(Cl)n1 CC1(C)CCC1C(=O)NC1CC(NC(c2ccn(C3CCC3)n2)=O)C1 N1(C(C(CC)SC)=O)C(C)C2CC1C2NC(=O)CNC(C1CCCC1)=O C1(NC(C2(CC)CC2(F)F)=O)CC2CCC(C1)N2C(=O)C1=C(C)CCCC1 C1(NC(C2C3(CN(Cc4ccc(C)cc4)C3)C2)=O)=CN=C(O)CN=C1C c1(C(c2n(CCCSC)nnn2)NCCOCCF)cccc(Br)n1 N1(C(c2c(C(=O)OC)scc2)=O)CCCCC(CNC(c2coc(CO)c2)=O)C1 C1(OCC)CN(C(=O)CC#N)CC1NC(=O)OC(C)(C)C.C12SCCN1C2=O c1(C(C)(C)C)scnc1C(=O)N(CCNC(C1CCCN1C1CC1)=O)C1CC1 C1(C(=O)NC(CCCCNC(C(C)n2cccn2)=O)C)CC2(C1)CC(C#N)C2 C1(NC(=O)CCc2ccccc2)CCSC12CN(C(=O)C(C1CCOCC1)O)C2 C1(N(C(c2c(C)nc[nH]2)=O)C)CCN(C(=O)C(C)Oc2ccc(O)cc2)CC1 C(=O)(CCN=C1NCC2CC(N1)C2)NC.C1(OC(=O)NC)CC(=O)N(C(C)C)C1 CCCCC#CC(C)(C)NC(C1CC(O)CN1C(C1CCC(=O)N(C)C1)=O)=O Cc1cc(=NC(C)c2ncnn2C(C)C)[nH]c(=NCc2nccc(O)n2)[nH]1 C(CC(O)C(=O)NCC(CC1CCCC1)C(=O)NCC(c1ccccc1)C)SC N1(C(c2cc(C)[nH]c2C)=O)CCCC(CO)(NC(C2CCSC(C)C2)=O)C1 c1(CCC)occc1C(=O)NC1(C(N2CC(N(CC(C)C)C)C2)=O)CC1(C)C C#Cc1ccc(Cl)c(C(=O)NC2CC(n3ccnc3)C2)c1 c1(NC(C(C)C)C(=O)NC2(C)CN(C(=O)C(=O)NC3CC3)C2)c(F)cccc1F C(=O)(C(C1=NOCC1)N1CC(C)(C#N)C1)NCCCOC N1(C(C(c2scc(C)n2)C)=O)CCCC(C2CN(C(C3CCOC3)=O)C2)C1 c1(OCC(=O)NCC(CC)NC(c2cncc(F)c2)=O)cncc(Br)c1 C1(C(N2CC(C(N)=O)(CNC(CCC)=O)C2)=O)CCN(C)C(C)C1 C1(NC2CN(C(C(C)OC(CNC(CC)=O)=O)=O)C2)CC(N=[N+]=[N-])C1 C1(C(=O)NC(CC=C)(C)C)C(C)CCN1C(=O)C=Cc1cocn1 N1(CC=O)c2c(Br)cccc2CC1C.c1(NC)cccc(Cl)c1C N1(C(C2(C#C)CC2)=O)C2CCC(C2)C1CC(=O)Nc1ccc(Cl)cc1O Cc1cncc(C(=O)NC2CCCC(NC(c3ccccc3Cl)=O)C2)c1 Cc1ccnc(C)c1C(=O)NCC1CCCN(C(C2CC3C=CC2CC3)=O)C1 c1(C(C)=O)ccccc1C(=O)N(C1CCN(CCO)CC1)C c1(C(=O)NC2(C)CN(C)C(=O)CC2)cc2n(c1)CCCNC2=O c1(C(=O)NC)ccc(F)c(-c2cccc(NC(C3CC4CCC3O4)=O)n2)c1 CC1CC=C(C(=O)NC2CCCCC2NC(=O)COc2ccc(Cl)nc2)CC1 N1(C(c2ccc(OC)c(F)n2)=O)CCCCCC(Nc2ccccc2[N+](=O)[O-])C1 c1(NC(C2C(C(=O)Nc3ccc(C4CCC4)nc3)C2)=O)ccc(Br)c(F)c1F O=C(C#CC1CCCCO1)NCC1CN(C(c2cc(C(F)(F)F)cs2)=O)C1 N1(CC(=O)NC2(C)CCN(C(Cc3c(C)cco3)=O)C2)CCSC2CCCCC12 CCCC(C)(CCC)C(=O)NC1C2CC3C(C2)C13C(=O)NCC(C1CCC1)OC C(c1ccc2c(c1)COCC2)=CC(=O)NC(C1CC(NC(COCC)=O)C1)C N1(C(CCCCNC(c2cc(C)c(O)nn2)=O)=O)CC2(CCC1CO)CC2 C(=O)(C1=CCCCCC1)NC(CC(=C)C)C(=O)NC1CCCC2C1C2(F)F N1(C(CC2OCCC(C)(C)C2)=O)Cc2ccccc2C(NC(=O)CC2(C)CC2)C1 c1(CC(=O)NCC(CC=C)NC(=O)CC(C)(C)COC)ccc2[nH]ccc2c1 N1(C(C(C)OCCCC)=O)CC=C(C(=O)N(CC(C)C)C)C1 c1(OC)cc(CNC(Cn2cncn2)C(=O)O)cc(C#N)c1 C(C(C)(C)C(=O)NCC(C)NC(=O)CCSCC(c1ccccc1)=O)SC c1(C(=O)NCCC2CC(OC)CN2C(C2CCOC2)=O)c(F)cc(Cl)cc1F C1(CNC(C(CC=C)C)=O)CC2(CCOCC2)CN1C(=O)C(F)=C1CCCC1 c1(C(=O)NC(C)CNC(=O)CCn2cc(Cl)cn2)ccc2nc(O)oc2c1 C1(C(=O)OCC)COCCN1C(C1CC1(C)C)=O.c12scnc1N2 C1(NC(c2cnc(CC)s2)=O)CC2(C1)CC2NC(c1cn[nH]c1)=O S(=O)(=O)(c1ccc(NC2CN(C)CC2O)cc1Br)N1CC(F)CC(C(C)C)C1 c1(OCCOC)ccc(NC(=O)C(N2CCCC(c3cncnc3)C2)=O)cc1 N1(C(CC2CC(N(C)C)C2)=O)CCOCC1C(=O)NCC1CCCCO1 Cc1cc(Cl)c(Cl)cc1CN(C1CN(C(c2c(C)cccc2C)=O)C1)C Cc1ccc(S(=O)(=O)C2(C(=O)NC3CCNS3(=O)=O)CCCC2)cc1 C1(CN(C)CC)CN(C(C2CCCCCCC2)=O)CCN1C(=O)Cc1cnc[nH]1 c1(C(N(C2(c3cc[nH]n3)CC2)C)=O)c[nH]nc1CNC(=O)CC1OCCO1 C1(NC(C2CCCN(c3nccs3)C2)=O)CCC2(CCNCC2)C1 c1(CC)noc(C(N2CCOCC2CN(C)C(C2(COC)CCCC2)=O)=O)c1C Cc1cc(C)c(C(=O)NC(C2CC2C(=O)NC(C)Cc2nn[nH]n2)C)s1 CCCC(C(=O)N1CCC(CNC(c2cccc3scnc23)=O)C1)C(C)C C(=O)(C#CC1(C)CC1)NCCN(C(C(c1ccccc1)SC)=O)CC1CC1 CCC(CN(C)C)CC(=O)NCC(CNC(c1nc(C(C)C)oc1C)=O)OC C(CCCCC(=O)N(C(C)CCNC(c1cn(C2CCC2)nn1)=O)C)=CC CC(C)CC(C(=O)NCC1CC2(CC2)CN1C(c1cc2n(c1)CCC2)=O)C(N)=O C(=O)(C(C)CS(C)(=O)=O)NC(C1N(C(c2cncc(CC)c2)=O)CCC1)(C)C N1(C(CC(=O)N(C)C)=O)CCC(C2(NC(c3c(F)cccc3Cl)=O)CC2)C1 N1(C(CCOCCOCC)=O)CCC2(CCN(C(c3ccc(C#N)[nH]3)=O)C2)C1 N1(c2nnc(CC)o2)C(CNC(=O)C=Cc2cocn2)CC2COCC12 c1(OCCC(=O)N(C2CC2)CC2CCNC2)ccccc1Cl c1(C(=O)NC2(CC=C)CCN(C(c3cc(C)c(Cl)s3)=O)C2)cccc(F)c1F c1(CC)noc(C)c1C(=O)NCC1(F)CC(CNC(C2CC2(C)Br)=O)C1 C(=O)(C1CCCn2ccnc21)N1C2(CNC(Cc3cc(C)no3)=O)CCC1CC2 Cc1nc2ccccc2n1NC(=O)NC1CCc2c[nH]nc2C1 CC1(C)CC(N=c2ccn3nccc3[nH]2)CN(c2nc3cccc(F)c3s2)C1 C(C)(C(=O)N1CC(c2ncccn2)C1)(N(C(COCCCN(C)C)=O)C)C1CC1 c1(CNC(N2CCOC(C(C)C)C2)=O)cc(F)cc2c1CCC2 c1(C(=O)NC(C)C(C)NC(=O)C=Cc2ccccc2)ncc(Cl)cc1Cl c1(OC)ncnc(OC)c1C(N1CC(C(C)NC(C2CCCCC2(C)C)=O)C1)=O CP(C)(=O)CC(=O)NCC1(NC(=O)NCCCCC2CCCOCC2)CCCC1 CC1(C(=O)NC2CC3CCC(C2)C3=O)CC(c2ccccc2Cl)=NO1 c1(C(N(CCN(C(c2ccc(C)nn2)=O)C(C)C)C)=O)cc(F)cc(Cl)c1N c1(C(C)C)cc(C(=O)NC2CC(O)(CNC(=O)C(F)=CC3CC3)C2)on1 c1(CC(=O)N(CCNC(C2C(OC)CC2)=O)C)cccc(C)c1Br c1(N(C(C(c2csc(C)c2)NC)=O)Cc2ccc(C)cc2)ccc(F)cc1 c1(COC(C(C)OC)=O)cc(=O)n2c(n1)CCCC2 c1(C(NC(=NCCCC)NCCCF)C)cnc2c(C)cccn12 C#CC1(C)CCCN(C(=O)C(C)(C)CN(C(=O)C(C)S(N)(=O)=O)C)C1 n1(CC(=O)NCCC2CCC(N(C(=O)CC3CCCCC3)N)C2)nnc(=O)[nH]1 c1(C(=O)NCCCCCCN(C(=O)CC2CCC(F)(F)C2)C)ccc([N+](=O)[O-])s1 CC1CC(NC(c2occ3c2CCC3)=O)CN(C(=O)Cc2cnns2)C1 O=C(NN=c1cc[nH]cc1Cl)c1n[nH]c2nn(CC(F)(F)F)cc12 C1(CC(=O)NCC=CCNC(C2C=CCCC2)=O)COCCO1 C1(F)(CNC(C)=O)CCC(CNC(=O)C(C)C2CCCO2)C1.n12ccnc1S2 C1(CCN(C(=O)CC2C=CCC2)C)CCCCN1C(c1ccoc1Cl)=O C1(C(N2CCC(O)(C(C)NC(c3coc(Cl)n3)=O)C2)=O)CC2C(C1)C2(C)C C1(COC)CCC(NC(=O)CC2CCCN2C(=O)CC2CC(SC)C2)CC1 c1(NC(C(C=C)C)=O)cccc(NC(=O)Nc2ccc(Cl)cc2)c1 C1(NC(c2c(C)nc[nH]2)=O)CCCCC1C(=O)NCC1(O)CCOC1 O=C(CCCCc1ccccc1)NCC(O)CCNC(C1CC1C(F)(F)F)=O C1(CNC(=O)C(O)C2CC2)CC2CCCCC2N1C(=O)CCC1CCCOC1 c1(CN=c2scc(-n3cnnc3)[nH]2)cccn2c(O)nnc12 C1(NC(c2cccc(CC)n2)=O)(CC)CCCN(C(C2CCC2)=O)C1 N1(C(c2n(CC)nnc2)=O)CCC2CCN(C(=O)C=Cc3nccs3)C2C1 C1(C2CN(C(C3CCO3)=O)C2)(NC(c2c(C)nc(-c3ccccc3)o2)=O)CC1 CCCCC(=O)OC1CC(NC2(C3CCCCO3)CC2)C1 C1(NC(c2ncc(C)[nH]2)=O)CCN(C(=O)C(=O)NCC2CC2(F)F)CC1CO C1(C(=O)NCCCS(C)=O)COCCC1NC(=O)Cc1nccn1C C12(C(=O)NC3CCN(C(c4c(N)c(Cl)ncc4)=O)CC3O)CCCN(CCC1)C2 c1(CN(c2nnc(-c3ccccc3)s2)CCN(C)C)ccc(Cl)cc1 c1(C(N(C2CCC(NC(CCC3C(C)C3)=O)CC2)C)=O)cn2cc(Cl)cnc2n1 C(=O)(C1CCc2c[nH]nc21)NC(CCC=C)C(=O)NCc1ncc[nH]1 C1(CNC(=O)C(N2CCC(C3CC3)C2)=O)CCC2(CCCCCC2)O1 N1(C(C(C)OC2CCCC2)=O)CCOC(CNC(=O)CCNC(=O)C(C)(C)C)C1 Cc1cc2c(cc1C)C(C(=O)NCCCCC(C)NC(C1CCCSS1)=O)CO2 C1(C(=O)OC)CCC1(C)C(=O)N(CCCNC(=O)C(C)CC)CC1CC1 C1(C(CC)C(=O)N(CCCN(C)C(c2ccnn2COC)=O)C)CCC(C)CC1 C(=O)(C(C)C(CC)CC)N(CCN(C(=O)Cc1ccco1)CC)CC N1(C(C(=Cc2ccco2)C)=O)CCN(c2ncnc(O)c2Br)CC(O)C1 CCCN(C1Cc2ccccc2C1)N1CCCC(OCc2ccc(OC)cc2)C1 CC(C)C(F)(CNC(=O)CC1OCCCO1)C(=O)NC(C)Cc1cccs1 N1(C(CC2(OC)CCC2)=O)CC2(CCCC2)C1C(=O)NC1(c2n[nH]c(C)n2)CC1 c1(C(N2CCC(CC)CC2C(N2CCC(C3CC3)C2)=O)=O)cccc2ccccc12 N1(C(C=C=C(C)C)=O)CCCC(C)C1CNC(c1cn(C)ccc1=O)=O N1(C(c2cccc(C(C)C)n2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 N1(C(c2c(Cl)ccc(OC)n2)=O)CC2CC(C1)N(C(=O)C(CO)N(C)C)C2 Cc1cc(N2CCN(C(=O)CCN3CCCCC3)CC2)cnc1O N1(C(C2CC(OCC)C2)=O)CCCOC(CNC(=O)C(c2ccccc2)C)C1 N1(C(C(C)CC(F)F)=O)CC2COCCC2(NC(c2ccc(Cl)cc2Cl)=O)C1 C(c1ccsc1)=C(C(=O)NCC(CC)NC(C1(N2CCNC2=O)CC1)=O)C C1(OCC)COCCC1CC(=O)NCC(C)N(C)C(c1ccoc1Br)=O c1(C(N2CCN(C(C(=O)NC(C)C)=O)C(C)C2C)=O)nnc(O)c2ccccc12 c1(NC(C2COCCN2C(c2c(F)ccnc2Cl)=O)=O)ncc([N+](=O)[O-])cc1Br C(CN=c1ccnc(C(C)C)[nH]1)C1CC(C)N(C(=O)CN(C)C2CC2)C1 C1(NC(c2scc(C)c2C)=O)CCC2(CCN(C(c3cncc(N(C)C)c3)=O)C2)C1 C1(CNC(C2N(CC)CCCC2)=O)CCCC12CCN(C(=O)COC(C)C)CC2 c1(NC(=O)CCN2CCSCC2)cccc(OC(F)F)c1Br CC1(C)CC(C#N)(CNC(=O)CC23CC(CN2C(C2CC2(C)C(F)F)=O)C3)C1 c1(CNC(C2CCS(=O)(=O)C2)C2CC2)ccnc(Br)c1F c1(CC)cccc(F)c1C(N1CCC(C)C1CNC(=O)C(C)(C)c1cccs1)=O N1(C(C(N2CCN(C)CC2)(C)C)=O)CCCC(NC(c2ccncc2)=O)CC1 N1(C(c2ccncc2O)=O)CC2(C(=O)NCC3(CO)CC=CC3)CC1CO2 C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C)N(C(=O)Cc1cc(F)cc(F)c1)C O=C(C1=CCCC1)NCC=CCNC(=O)Cc1cccc(O)c1 c1(C(N2C(CNC(c3c(SC)ccs3)=O)CC(C)(C)C2)=O)cc2ccncc2[nH]1 Cc1cc(Br)cnc1C(=O)N(C1CC1)CC1CCN(C(C23CCCC2C3)=O)C1 C(C)(C(=O)NC1CCCCN(C(=O)CCc2cncn2C)C1)(C(C)C)OC CC(C)(C)C1=NOC(C(=O)NC(c2ccccc2F)CNC(=O)C2=CCCC2)C1 Cc1cccnc1C=CC(N1CCC(NC(=O)CCc2cn(C)cn2)CC1C)=O N1(Cc2n(C(F)F)cnc2)CCn2ncc(-c3nn[nH]n3)c2C1 N1(C(CN=c2c(C(=O)OCC)cc(Cl)n[nH]2)=O)CCC(C2CCCC2(C)C)C1 CC(C)C(C(=O)NC1(C)CN(C(=O)C(C)(C)O)C1)N(C)C N1(C(C2C(C)N(C)CC2)=O)CCOC2CN(C(=O)Cn3cnc(C#N)n3)CC12 C(CCCCC(=O)NC1CCN(C(c2cnc(OC)c(Cl)c2)=O)CC1C)OCC C(=O)(C1=CC2(CCOCC2)C1)NCC1C(NC(CC=CCC)=O)CCCC1 C1(C)(CC)C=C(C(=O)NC(C(=O)N(C)CC)C2CCC2)C1 CC1(C#CC(=O)NCC2CN(C(=O)CCOc3cc(Cl)cc(Cl)c3)CCO2)CC1 C1(N(C(C(=O)NC2(C)CC2)C2CC(CC=O)C2)C)CCCCC1.N1(CC)CCCC1 C1(CC(=O)NCC2(CNC(c3csnc3Cl)=O)CC=CC2)CC=CCC1 C(=O)(C(CC)C(=O)NCC1CCC1C(=O)NC(C(O)C1CC1)C1CC1)OCC N1(C(COC2(C)CCC2)=O)CC2(CC(C(=O)N(C3CCC3)C3CC3)CO2)C1 N1(C(C)=O)CCCC(C)C1CNC(=O)CCc1ncc[nH]1 c1(OC)ccc(CCC(=O)NC(C)CN(C(=O)CC2CCCCO2)C)cc1OC C1(C(N2CCC(N(C(=O)CC3C=CC(COC)C3)CC)C2)=O)CC2OC1C1CC21 N1(C(C(CCC)N(C)C)=O)CC2CC1CN(C(=O)CC1CSCCO1)C2 C1(C)(C(N2CCCC(CNC(C(C(=O)NC)(C)C)=O)C2)=O)CCC(C)C1(C)C N1(C(C=CC=CC)=O)CCN(C(=O)Cc2ccc(SCC)cc2)C2(CC2)C1 Cc1ccc(S(=O)(=O)N(C(C)C)Cc2ncc(-c3ccccc3)o2)c(C#N)c1 C1(C(=O)NCC2CN(C(C3CCN(C(=O)OC)CC3)=O)C2)CCS(=O)(=O)C(C)C1 N1(C(C2(SCC)CC2)=O)CCCC(N2CCC(NC(c3n(CC)ncn3)=O)C2)C1 Cc1cccc2c(=NCCC(C)N3CCCC3)[nH]c(=N)[nH]c12 C1(Cn2cc(CC=C)nn2)CCN(CC(=O)NCc2csnc2C(=O)O)CC1 N1(C(c2c(C)c[nH]n2)=O)CCC2(CCN(C(=O)CCCC(C)(C)C)CC2)C(C)C1 N1(C(C2C3CN(C(=O)Cc4ccc(F)cn4)CC32)=O)CC2CCC(C1)O2 c1(C(N(CC(CN(C(C(CC)F)=O)C)O)C)=O)cc(OC)ccc1[N+](=O)[O-] c1(CNC(Cc2cc(C)ns2)=O)cccc(CNC(C2CCS(=O)(=O)N2)=O)c1 c1(C(N(C2CC(NC(C3C(C)C3C)=O)C2)C)=O)cc(N(C)C)c2ccccc2n1 c1(NC(CN(CCC)C)=O)cccnc1CNC(C1(CO)CC1)=O C12CCCN(C1)Cc1cn2nn1.CCC(CO)CO.C(C)(C)(C)S N1(CC(=O)NCC2C3CN(C(c4cc(C)sn4)=O)CC32)CCc2ccccc21 C1(C(=O)NCC(COC)(C)CO)CCOCCN1C(=O)Cn1ncnn1 c1(C(N2CCC(C)(O)C2)C(=O)N(CCCC(=O)OCC)C2CC2)ccccc1O C(c1ccncc1)=CC(=O)NC12CC(CNC(C(C)OCC(F)(F)F)=O)(C1)C2 CCCC(C)(O)CC(=O)NC(CC(=O)NCCc1cnc(C)cn1)C1CC1 c1(C(=O)NCC2C3CN(C(C(CC=C)(C)C)=O)C2C3)c[nH]c2cccc(F)c12 C1(C)(CNC(c2c(CC)con2)=O)CCCN(C(c2nn(C)cc2C(C)=O)=O)C1 C1(NC(CC2CCC(=O)NC2)=O)CCS(=O)(=O)C12CN(C(=O)CCC[N+](=O)[O-])C2 c1(N2CCC(CCC(=O)NC)CC2)nc(N2CCC(S(N)(=O)=O)C2)nc2c1CSC2 c1(-n2c(-c3ncc(OCC)nc3)nc(C(C)COC)n2)ccc(Br)c(C)c1 C12(C(NOCC(=O)OC)=O)COCC1CN(C(C1CC(C)=NO1)=O)C2 N1(C(C2(C)CC=CCC2)=O)CCCC(C(=O)N(C2CC2)C2CC2)CC1 C(=O)(CC(C)(C)F)N(C)CC1C(NC(c2cc(OC)ns2)=O)CCC1 C1(NC(C2C(C)C2)=O)CCN(C(c2cc(Br)sc2Cl)=O)CC1F C(=O)(C1CCCc2nc(C)[nH]c21)NC1(C)CN(C(c2cc(C)nn2C2CC2)=O)C1 O=C(CCC1=CCCCC1)NCC(C1CC1)NC(c1ccsc1)=O C1(C(=O)NC(C2CCN(C(c3cnc(SC)n3C)=O)CC2)C)COC2COCC12 c1(OC)cc(F)cc2[nH]c(NC(N3CCC4CN(C5CCC5)CC4C3)=O)cc12 c1(CC(CCOC(CSc2nnc(C)o2)=O)=O)ccc(C)c(C)c1 C1(C(=O)NCC2C3CN(C(c4ccc(C)nc4C)=O)C2C3)CC2CSCC(C1)C2 c1(SC)ccc(-c2ccnc(CC(N3CCOC(NC(=O)C4CC4)C3)=O)c2)cc1 N1(C(C2C(C)OC(C)C2C)=O)CC2(C)CN(C(=O)C3=CCCOC3)CC2(C)C1 N1(C(C)=O)CCC(N=c2[nH]c(CCN3CCN(C)CC3)nc3c2CCC3)C(F)C1 c1(OC)ccc(CCC(N2CC(C(F)(F)F)C(CNC(=O)C(C)SC)C2)=O)cc1 C(C(C)C(=O)NC1COCC1NC(c1c[nH]nc1-c1ccccc1)=O)OC(C)=O c1(OC)ccc(C(=O)NCC2CN(C(=O)C=CSC)CC2C(F)(F)F)c(C)c1 C12(N(C)C(C3(CC4CC4)CC3)=O)CC1CN(C(C1(CNS(C)(=O)=O)CC1)=O)C2 N1(C(CCOC(CC(C)C)C)=O)CC(NC(=O)C=Cc2cc[nH]c2)C2(CCC2)C1 N1(C(c2c(CC)occ2)=O)CCN(C(=O)C(C)(COC)COC)CC1C N1(C(c2nc(C)c(C)[nH]2)CC)CCC(O)(c2cn(-c3cnn(C)c3Br)nn2)CC1 CC1CCCN(C(=O)C=Cc2cnn(C)c2)C1CNC(=O)CCCCC1CC1 C(=O)(C(O)CCCNC(=O)C(O)C(F)(F)F)N(C1CS(=O)(=O)C1(C)C)C CS(=O)(=O)c1ccc(F)cc1C(=O)NCCCN(C(=O)C1=CCSC1)CCO c1(N2CCC(C=C)CC2)[nH]c(=NCc2c[nH]nc2C2CCCCC2)nc2scnc12 n1(CC(N2CC(CC)N(C(=O)CCC3(C)N=N3)CC2)=O)ccc2c(C)cccc12 c1(C(N(CC(=O)O)CC)=O)ccc(N2CCOCC2)nc1C C(=O)(CCCCCCCC1CC1)NCC1CC(CNC(c2n(CC)cnn2)=O)C1 C1(C2CCN(C(C3CCC(O)C3)=O)CC2)(NC(=O)CCCCC(F)F)CC1 C1(C(N(CC(C)NC(c2c(C)[nH]nc2C(F)F)=O)C)=O)CCCC1S(C)(=O)=O c1(CC)nn(C)c(CC)c1C(=O)N(C)CC1CCCN1C(=O)CN(C)CC C1(CC)COCCN(C(C2(C)CC3CCC2O3)=O)C1.C12CCC1NC2=O C1(CNC(c2c(C3C(C)C3)noc2)=O)CN(C(=O)CC(C)(F)F)CC12CC2 C(CCN=c1cc(C#N)nc(C(C)C)[nH]1)N(C(CS(CC(C)C)(=O)=O)=O)C c1(C(=O)NC2CCC(NC(=O)COC3CCOCC3)CC2)ccnc2c1CCC2 CCCCCCCC(=O)N(C1CC(NC(C2CC(F)(F)C2(C)C)=O)C1)C CCC(CC(=O)NC1(C)CCN(C(=O)CCn2ccnc2C)C1)C(C)(C)C N1(C(C(CC)(C)C(N)=O)=O)CC2CCN(C(c3ncn4cc(Cl)ccc34)=O)CC2C1 c1(CC)ccc(O)c(C(=O)N(CC(CC)NC(c2cccc(C)c2F)=O)C)c1 Cc1ccc(CC(N2CCN(C(=O)CC3CCOC3)C3CC23)=O)c(Br)c1 C1(C(=O)O)C(N)CCCN1Cc1ccc(N2CCNCC2)o1 CC1CN(C(c2cc(F)c(Cl)cc2Cl)=O)CCCN1C(c1c[nH]nc1F)=O Cc1n[nH]c(C)c1CC(N1CC(C(C)NC(=O)CCCc2cccnc2)C1)=O c1(C(=O)NC(C(C)(C)C)Cl)ccc(OCC(=O)NC2CC2)cc1 c1(CNC(=O)NC2CC(CO)C3CC23)nccc(Cl)c1O C(=O)(CS(=O)(=O)C(C)C)NCCC1(O)CCN(C(c2ccc(COC)[nH]2)=O)CC1 C1(CC(N2C(C)CC(CNC(C3(C)C(C)CCC3)=O)C2)=O)CN2CCC1CC2 Cc1c(C(=O)NC2CN(C(=O)CN(C3CCSC3)C)C2)cc(N)cc1O CCC(CN(C)C)CC(=O)NC(C)C(=O)NCCS(N)(=O)=O CCCC(C(F)(F)F)NC(C1CCCN(C(=O)CCOCC2CC2)CC1)=O Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)CNC(c1ccco1)=O Cc1ccc(C(=O)N(C2CN(C(=O)CCCC(C)(F)F)C2)C)c(N)c1C C12(C(=O)NCC(C)CNC(=O)C(c3ccc(Cl)s3)C)CC3CC1C2C3 Cc1ccc(CC(N2CCN(C)CC2CNC(=O)C(=O)NC2CC2)=O)c(F)c1F C(=O)(C(C)C(C)(F)F)N1C(CCSC)C=CC1.c12ccc(cc1)-c1cn(nn1)C2 N1(C(C=C(C)Cl)=O)CC2CCC(C1)N(C(c1cncc(F)c1C(F)(F)F)=O)C2 C#CCCCCCCC(=O)N(CC(N1CCC2(CC1)CC2C#N)=O)CC#C C1(NC(COC2CCCC(C)C2)=O)CN(C(=O)CS(N)(=O)=O)C(C)(C)C1 C1(CCCCNC(N2CCC2CO)=O)CCCN(C(C2CCOC2)=O)C1.C1COO1 CC1(C)CC(CCNC(=O)CC2(NC(=O)CCc3cccn3C)CC2)CO1 c1(N2CCOCC(CNC(CC(C)SC)=O)C2)ncnc2c(C)csc12 CC12CC(C(N3CCN(C(C4CC5CCC(C4)S5)=O)CC3)=O)(C1)C1(CCC1)O2 c1(C(=O)NCC2(F)CC(NC(Cn3ncn(C)c3=O)=O)C2)cn2cccnc2n1 N1(C(C(COC)(C)O)=O)CC2CC(NC(c3ccc(OC)nc3Cl)=O)CC2C1 N1(C(C2CCCC(NC(=O)OC(C)(C)C)CC2)=O)CCOC(C(=O)O)C12CCC2 c1(CCNC(=O)NCC(=O)NCc2ccccc2)ccc(Br)s1 c1(C(=O)NCCN(C(c2ncc(C)cc2C)=O)C)cc(N)c(F)c(F)c1F C=CCC(CNC(=O)CCNc1ccccc1)NC(=O)C=C(Cl)Cl c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCC2(C)C(C)C)=O)s1 c1(OC)cnc(NC(=O)COC(=O)CC(C)SC)nc1O N1(CCC(=O)NCc2cc(C#C)cc(Br)c2)CCn2cc(C)nc2C1 C1(C)(CC)C=C(C(=O)NC2COCC2NC(c2ccc(F)cc2)=O)C1 C1(C(=O)NC(CC=C)CNC(=O)C(C)CN(C)C)CCN(CC(F)F)CC1 C(CCC(C)C(=O)NC1CCCC(CNC(=O)CCC=CC(C)C)C1)OC CCC(CNC(=O)CCCc1nc(-c2ccc(C)cc2C)no1)CC(F)F C1(C(N2C(CN3CC(CN(CCC)C)OCC3)CCC2)=O)CS(=O)(=O)CC(=O)N1 C1(CNC(CCNC(=O)CO)=O)CCCN(C(=O)CN2CCCNC2=O)C1 Cc1cc(C(=O)NCC2CC3CC3N2C(=O)COCCCF)n(C)n1 C1(C(=O)NCCC#CCO)(CNC(c2ccc(CO)s2)=O)CC2(CC2)C1 Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(c2sccc2C(F)F)=O)cc(O)n1 C1(C(C)NC(=O)CC(=O)NCC2CCC2CCC(C)(C)C)CC(C)(C)C(C)(C)C1 Cc1cc(NC(C23CC2CN(Cc2[nH]c(C)nc2C)C3)=O)cc(Br)c1 c1(CNC(=O)CSC2(C(F)(F)F)CC2)cscn1 c1(C(N(CC(C)NC(c2cc(CSCC)on2)=O)C)=O)n[nH]c2c1COCC2 CP(C)(=O)c1cnc(C(=O)Nc2cc(Br)cc3c2OCCC3)nc1 C(C(C)N=c1cccc(S(=O)(=O)N2CCC3(CCC(C)CC3)C2)[nH]1)OC(C)C N1(C(CCC)=O)CC2(CC(C(=O)NC(C)CCC(F)(F)F)CO2)C1 N1(C(c2n(C(C)C)ccn2)=O)CC2CCCC(CNC(=O)C(F)=CCCF)(C2)C1 N1(CC(CCNC(=O)OC(C)(C)C)(C)O)Cc2nc[nH]c2C1 C1(NC(C2(C)CS(=O)(=O)C2)=O)CCC2(CCCN(C(c3cc(Cl)cn3C)=O)C2)C1 C#Cc1cncc(NC(=O)C(CCF)NC(=O)Cc2cn(C)cn2)c1 c1(C(N2CC(C(C)NC(=O)Cn3cnnn3)C2)=O)cccn2c(O)nnc12 CC(C)C(F)C(=O)NCC(C1CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1)(C)C c1(C(=O)NC(C(C)OC)C(=O)NCC2(CC3CC3)CC2)ncc(C)cc1C C1(NC(c2cnn(CC)n2)=O)CCN(C(C2CC(C)OC(C)C2)=O)CCC1CO C(=O)(CC(O)CC(C)(C)C)N(CC(=O)N(C(C)C(=O)Nc1cc(C)on1)CC)C C1(CNC(=O)NC2(C(F)(F)F)CC(O)C2)CCC2CC2C1 C1(CNC(c2scc(OC)c2)=O)CCCCN(C(=O)Cc2cc(C)cc(F)c2)C1 c1(CC(=O)NCC2(F)CN(C(CC(CC)C3CC3)=O)C2)ccc(CO)cc1F c1(C(N2C(CNC(c3c(C)ccs3)=O)CC(F)C2)=O)cc2c(Cl)cncc2s1 C1(C(=O)NCC=CCNC(CN(CCCOC)C)=O)COCC(=O)N1C(C)C C(CCC(C)C(=O)NCCCCCN(C(=O)CN1CCC(F)(F)C1)C)OC C(=O)(CCC(F)(F)F)NCCC1(C)CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(NC(CC(C)(C)c2ccccc2)=O)COC2CN(C(=O)Cc3cnc[nH]3)CC12 N1(C(Cc2ccc(C)o2)=O)CCC(C)N(C(c2n[nH]c3c2COC3)=O)CC1 c1(C(N(C)CC2(NC(C(C3CC3)OC)=O)CC2)=O)ccc(Cl)cc1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)C(C)Cc3ccccn3)cc2o1 c1(C(N2CCC(NC(C3(C)CC3)=O)CC(F)C2)=O)ccc2[nH]nc(Cl)c2c1 N(C(=NCCC1COC(C)(C)OC1)NCCF)CC1C(C(=C)C)OCC1 C12(C(=O)NCC(CCNC(=O)C3CC3)O)CCC(CO)(CC1)CC2 c1(NC(=O)CN2CCC2C2CCOC2)ccc(F)c(F)c1F C1(C(C)N(C)C(c2occc2CNC(C2(CO)CCCO2)=O)=O)CCOCC1 c1(N2CCN(C(C(c3nc4ccccc4o3)C)=O)C(C)C2)ncc2ccsc2n1 N1(C(c2c(C)n[nH]c2C)=O)CCCC(C(=O)NCc2scnc2C)CC1 C1(CN(C(C2(COC)CCC2)=O)C)CCCN1C(=O)COC1CCCC1 c1(CC(=O)NC2C(CNC(CC)=O)C2)sc(C)nc1C.C1C(=O)N1 C1(CNC(CCCOCC)=O)(NC(=O)Cn2cc(CN(C)C)nn2)CCOCC1 CN=c1[nH]nc(CC(=O)NC2CC2NC(c2ccc(SC)cc2)=O)s1 C1(O)(CN(C)C(C2CC(=C3CC3)C2)=O)CCCN(C(=O)CCCF)C1 C(=O)(C(F)CC(C)C)N.C12CCC(CC1)CNC(=O)c1csc(c1)C(=O)N2.COC N1(C(C=COCC)=O)CCC2OCCN(C(c3cncnc3)=O)C2C1 N1(C(CCC2(C#N)CCC2)=O)CC2CCC2(C(=O)NC2CC(CF)C2)C1 c1(C(=O)NCC2CN(C(C(n3ncc(C)c3)C)=O)CC2C)ncccc1N=[N+]=[N-] C1(NC(C(OC)OC)=O)CN(C(=O)CC(=O)N(C)C)CC1C CC1CCN(C(C2CC3(CCN2C(c2cc[nH]c2)=O)CC3)=O)CC1(F)F c1(C(N2CCC(C)(CNC(c3cc(F)c[nH]3)=O)C2)=O)ccc(O)c2c1CCCC2 c1(C(N(C2CCCN(C(CC)=O)C2)C)=O)cccn2c(O)nnc12 C1(C(N2CC(OC)(CNC(C3CC(C)OC(C)C3)=O)C2)=O)CCS(=O)(=O)C(C)C1 C1(C(N2CCCC2(C)CO)=O)(NC(CC(=O)OCC)=O)CC(F)(F)C1 Cc1nc(C(C)(C)C)sc1CC(=O)NCCSC(F)F c1(C(N2CCC(NC(C3CC3CF)=O)CC2)=O)ccn2ccccc12 c1(C(N(C2CCN(C(c3cc(CCC)n(C)n3)=O)C2)C)=O)[nH]cc2c1CCCC2 c1(C(=O)OC)cc2c(N3CCC(NC(=O)COC(F)F)CC3)[nH]cnc-2n1 Cc1ccc(F)cc1C(N1CCCC(C(C)C(=O)NC2CCCCCCC2)C1)=O CCCC(C(=O)NC1CC1NC(c1cnn(CCOCC)c1)=O)NC(C)=O N1(C(Cc2ccn(CC)n2)=O)CCC(CC(N2CCC2(C)C)=O)C1(C)C S(=O)(=O)(c1cc(C(=O)NC2CC(CCNC(C3(C)CCC3)=O)C2)c(C)o1)NC C1(NC(CN(c2ccccc2)C)=O)CCOC2(CCS(=O)(=O)CC2)C1 Cc1nc(O)nc(S)c1C(N1CCCC1(C)CNC(=O)C(c1ccccc1)O)=O C1(NC(C2CCCN(C(C3CCC(C)NC3=O)=O)CC2)=O)CC2C=CC1C21CC1 n1(CC(=O)NC(CC)CNC(C(CC)(F)F)=O)ncc(C)cc1=O C(=O)(C1OCCc2cc(O)ccc21)NC(CCCNC(c1c(C)[nH]cc1)=O)(C)C CCCCC(C)C(=O)NCC(CNC(c1ccc(Br)cc1Cl)=O)CO C12(C(=O)NCC(CNC(C(C(C)C)n3cccc3)=O)C)CC(C)(C1)OC21CCC1 CC1(C)COCC1C(=O)NCc1ccc(C(=O)NCCCC(F)F)cc1 c1(C(=O)NC2CCC(NC(=O)Cc3cnn(C(F)F)c3)C2)cc(O)ccc1F C1(C(N(C)CCC2CC2)=O)CC(CNC(=O)COC2CCC2)C1 Cc1cc(F)c2cc(-c3nc(C(C)Sc4cccc([N+](=O)[O-])c4)nn3C)[nH]c2c1 c1(C(=O)NC2C(C)CN(C(=O)C(C)(O)C3CCC3)C2)cc2c(ccn2C)[nH]1 N1(C(CSCC=C)=O)CC2CC2(CNC(C2CC(C(F)F)C2)=O)C1 N1(C(c2ccsc2Cl)=O)CC2CCC2(C(=O)NCC(CO)C2CC2)C1 C(=O)(C(CO)C(F)(F)F)N1C(CNC(c2cncnc2C2CC2)=O)CC2CC21 C1(C(=O)NCC(COC)NC(C2(OCC)CC2)=O)CCOC(C)C1 C1(NC(c2n[nH]cc2CNC(c2ccsc2SC)=O)=O)CCN(C(=O)NC)C1 c1(SCCNC(=O)NCCN(OC)C)cccc(Cl)c1 CCCCC(C)(F)C(=O)NCC1CC12CCN(C(=O)CC(=O)OC(C)(C)C)CC2 Nc1cc2c(cc1C(=O)NC(C1CCOC1)CNC(C1(O)CC1)=O)OCO2 N1(C(C2(CC)CCCN2C(=O)CCC=C(C)C)=O)CCOC2COCC12 C(=O)(C(C)(C)C(=O)N1CCC(CNC(=O)CC2CC3(CC3)C2)C1)OCC c1(C(=O)NC(C(F)N2CC(CCCCSCC)C2)=O)cccc(C(F)(F)F)c1O N1(C(=O)NC(c2scc(C(=O)OC)n2)C)CCOC(c2cccc(O)c2)C1 N1(C(C(C)(C)OC(C)C)=O)CCCC(CCC(=O)NCC(C)CC2CCC2)C1 C1(C(N2C(CC)CN(C(c3cc(C)c(N)cn3)=O)CC2)=O)CCn2ncnc2C1 C(CNC(=O)CCc1nccs1)(C(C)C(C)C)NC(c1ccn(COC)n1)=O Cc1nc(CC(=O)NCCC(C)N(C(=O)CC2CCCO2)C)c(Cl)s1 c1(C(=O)NCCO)ccnc(N)c1.C1(C(N)=O)(CO)CCCCC1.C12(CC1)N(C)C2=O c1(C(=O)NCC(CCC)NC(c2c(C)n[nH]c2C)=O)cc2ccnc(Cl)c2[nH]1 c1(C(N(C2CCCC2)CCNC(C2CCC3CC23)=O)=O)c[nH]c2ncccc12 C1(C(=O)NC(C2CCCN(C(c3cnc(S)[nH]3)=O)C2)C)CN2CCCN1CC2 S(=O)(=O)(c1c(OC)noc1C(C)(C)C)NC(=O)NCC1(F)CC(CC)C1 CC1CCN(C(c2cnsn2)=O)CC1NC(=O)CCn1cnccc1=O CCCCCCC(=O)NC(CCC1CCC1)C(N1CC(S(C)(=N)=O)C1)=O N1(C(CSCCOC)=O)CC2(CCN(C(c3cnc(O)c(F)c3)=O)C2)C1 c1(CC(=O)Nc2cn(CC)nc2)ccc2c(c1)CCCC2.N12CCOC(C1)C2=O C(C(C(=O)NCCCOCCOCCNC(=O)CCc1scnc1C)C1CC1)SC C1(CNC(C(C)SCC)=O)CC2(CO1)CN(C(c1c(Cl)nn(C)c1C)=O)C2 C(=O)(CC1=CCCC1)N(C)CC1CCN(C(C(CC)OC2CCCCC2)=O)C1 C(=O)(C#Cc1ccccc1)N1CC(C)(CC(N2CCC23CC(C(N)=O)C3)=O)C1 C1(CC(c2cn(C(Cc3ccccc3)CO)nn2)O)Cc2cc(F)ccc2O1 c1(COCC(=O)NCC(C)CNC(=O)Cc2cnsc2)cc(F)cc(F)c1 N1(C(C(c2cncnc2)C)=O)CC(C(N)=O)(CNC(=O)Cc2ccns2)C1 c1(C(=O)NC2CC(NC(C3(CCN4CCC4)CC3)=O)C2)cccnc1 C(c1ccc2[nH]ccc2c1)=CC(=O)NCC1C2CN(C(C3CC(=C)C3)=O)CC21 c1(C(N(CCCCNC(=O)C(F)CC2CC2)C)=O)cnc(O)cc1C(F)(F)F c1(C(=O)OCCSc2ccccc2)cc(O)ccc1C(F)F C(=O)(C1=Cc2ccccc2C1)NC1CC(C(=O)NC2CN(c3ccncc3)C2)C1 C(CCCC(=O)NCC12CC(CCO1)C2)NC(CCC1(C#N)CCC1)=O Cc1c([N+](=O)[O-])c(C(=O)NCCc2cnc(C3CC3)nc2)nn1C C1(c2cn(CCN(C(C)=O)CC)nn2)COCCN1C(=O)OC(C)(C)C C12(NC(C3C(C)C3C)=O)CCC1CN(C(=O)CCc1cc(Br)ccc1F)C2 CC1CN(C(C2CN(C(c3cccc(-n4cncn4)c3)=O)CCO2)=O)CC(=O)N1 C(=O)(C(CC=C(Cl)Cl)c1ccccc1)N1CCCC(C)(C(=O)O)C1 C(C)(CC(=O)N1CCC(CCNC(=O)Cc2cc(C(F)(F)F)n[nH]2)C1)OC C1(C(=O)NC2C(CNC(c3c(C)occ3)=O)C2)CCC12CCC2 C(CCCC(=O)NCC1(F)CC(NC(c2cnccc2Br)=O)C1)OCC C12(CNC(c3cc(CN(C)C)no3)=O)CC1CN(C(=O)CCOC1COC1)C2 c1(C(=O)NCC2N(C(CC(CCC)C)=O)CCCCC2)cc(F)c(N)cc1F n1(C(CC)C)nnnc1C(CC)(C1CC1)NCCOCC(C)C CCCC(CNC(=O)C(CC)CCOC)C(=O)NC(C(=O)NC)C1CC1 C(=O)(CCn1cccn1)NCC1(CN(C(=O)C=CCF)C2CC2)CC1 c1(NC(C2C(C(=O)Nc3nc(C)c(Br)s3)C2)=O)cccnc1[N+](=O)[O-] C1(NC(Cc2c(CC)cc(F)cc2)=O)CN(C(=O)CC2CC2)C2(CCC2)C1 N1(C(CNC(=O)OC)=O)CC2CC2(C(=O)NC(C)CCN2CCCC2)C1 Cc1nn(C)cc1CC(=O)NC1(c2cn(-c3nccs3)nn2)CCC1 c1(CC)ncncc1C(=O)NC12COC(CN=c3[nH]nco3)(C1)C2 C(=O)(CCCC(N)=O)NC1(C)CCN(C(Cc2c(C)cco2)=O)C1 C(=O)(C(C(=O)N1CC(CCCCNC(=O)C(F)C(C)C)C1)OC)OCC C#CC12CCC(C(=O)NC3CC(CNC(=O)C(C)(Cl)Cl)C3)(CC1)CC2 CCCC(CC)CC(=O)NCCC(F)Cn1cc(-c2ccc(C)cn2)nn1 c1(C(N(C(C)CNC(C2CC(N(C)C)C2)=O)C)=O)ccc2cc(O)ccc2n1 N1(C(c2c(C(C)C)ocn2)=O)CCC(F)C(NC(C2(C)CCN(C)C2=O)=O)C1 C1(NC(CC=CC=C)=O)(CO)CCCN(C(C2CCC3CC2CO3)=O)C1 N1(C(CSSC)=O)CCCC2CN(C(c3nnc(-c4ccccc4F)s3)=O)CC12 C=CC1CN(C(=O)CCn2c(C)csc2=O)CC1NC(C1CCCCCCC1)=O N1(C(c2c(C)nc(C)o2)=O)CCCC(C)(CNC(=O)C(c2ccccc2)F)C1 C1(N(C(=O)CN2CC3CC3C2)C)CN(C(c2cc(C(F)(F)F)nn2C)=O)CC1F CCCCC(O)C(=O)N1CC(NC(c2cncc(C(C)(F)F)c2)=O)CC1(C)C c1(NC(C)=O)ccccc1CC(=O)NC1CC1C(=O)NC1C(C)(C)C1(C)C CCC(C)C(C(=O)N1CC(OC(F)F)C1)NC(=O)Cc1cnsc1 c1(C(=O)N(C2CC2)CC2CCC3CC23)ncccc1NC(=O)CC(C1CC1)C1CC1 c1(C(N(CCOC)C(c2ccc(OC(C)C)nc2)C)=O)cnc(OC)c(CN)c1 c1(C(N2CC(C)C(NC(=O)CC(F)(F)F)C2)=O)ccc(O)c(O)c1O CC(C)(C(=O)N(C1CC2(C1)CC(O)C2)C1CC1)C(=O)N1CCOCC1.C(C)(C)C C12(NC(CC3C(C)C3)=O)CC(CNC(C3(CC4CC4)CCC3)=O)(C1)C2 N1(C(c2n(C)cnn2)=O)CCCCC1C1CCCN1C(=O)Cc1cccc(F)c1 c1(C(N(C2CCN(C(c3cc(C(N)=O)[nH]n3)=O)CC2)CC)=O)cc(Cl)c(Cl)[nH]1 CC(c1cccc(Br)c1)=CC(=O)NC1CN(C(C2(C)CCC2)=O)CC1(C)C C1(NC(c2n(C)ncn2)=O)CCC2CC1CN2C(C1CC12CC(C)(C)C2)=O C=CCC(CC=C)C(=O)NC1CCN(C(c2c[nH]c(=N)nc2CC)=O)C12CCC2 C(N=c1nc2ncn(C)c2c[nH]1)C1CCN(N(C2(C)CCCC2)C)C1 C1(COC)(CNC(C2CC23CCCC3)=O)CCCN1C(=O)CC12COCC(C1)C2 c1(OC)ccc(C2CSCCN2C(=O)CCCn2cccn2)cc1 C(=O)(CC(C)C(=O)N1CCN(Cc2cn(-c3ccc(F)cc3Cl)nn2)CC1)NC c1(C(=O)NCC2CC(NC(c3occc3C3CC3)=O)C2)ccc2[nH]nc(O)c2c1 C1(NC(c2cn(CC)nc2)=O)CN(C(c2nn(C)cc2N)=O)CC(C)(C)C1 CC1CN(C(c2sccc2Cl)=O)CCC1NC(=O)Cc1cnn(C(F)F)c1 N1(C(COCCCC)=O)CCN(C(=O)CC2CC(CC)=NO2)CC1C(F)F C1(C)(C(=O)OC)C=CCN1C(=O)CNC(C1CCN1C)=O CCCCC(C)CCC(=O)NCC1C=CC(NC(=O)CC2(CSC)CC2)C1 c1(OCCN(C)C)cccc(F)c1.C12COCC1C(=O)NC2 c1(C(=O)NC(CCCNC(C(F)=C(C)C)=O)c2ccccc2)ccc(=O)n(C)c1 N1(C(Cc2c(C)ocn2)=O)CCC2(CC1)CN(C(=O)C1=NOC(C)C1)CC(C)O2 c1(-c2cc(NC(N3CC(C)N(C)CC3)=O)on2)ccc2c(c1)OCCO2 N1(C(CC(C)OCC)=O)CCC(CC(=O)NC(C(C)OCCOCC)=O)C1 Cn1nnc2c(C(=O)NC3(CO)CCN(C(c4cccc(F)c4)=O)C3)ccnc12 c1(C(C)(C)OC)ccc(C(N2CCCC(NC(=O)CCC(C)C)C2C)=O)c(O)n1 N12CC(CO)CC1C2=O.C(C(F)C(=O)OC)N(C1CC1)C(C1(CC)CCC1)=O c1(C(N(CC(=O)NCC(COC=C)C)C(C)C)=O)conc1CC c1(CC(=O)NCC(C)(C)CCNC(C2CCOC2)=O)ccc2nsnc2c1 CC1(CCC(=O)NCC(=O)NCC(=O)NC(N)=O)CN(C(=O)CO)C1 C1(C(C(=O)NCC(C)NC(c2ccccc2OC(F)F)=O)C)CC(C2CC2)C1 C#Cc1cc(C(=O)NC2CC3CC2CN(C(=O)Cc2cscn2)C3)ccc1Cl CCC(CC(=O)N1CCN(C(c2cc(C)nc(O)n2)=O)C(CF)C1)C(F)F C1(C(N(CC(=O)NC(c2cncnc2)C)CC)=O)CCCC(C#N)C1 CC(C)CC(CNC(c1cn[nH]c1)=O)C(=O)NCC1(F)CCOCC1 CCCCC(CC(=O)NOCCN1CCCC1)NC(=O)CCCCN(C)C c1(C(=O)NCC(CCCC)NC(c2ccoc2CCC)=O)[nH]cc2c1CCC2 C(=O)(C(C)(CCC)CCC)N1CCC(NC(CCC#CC)=O)C(C)C1 N1(C(C(C)S(N)(=O)=O)=O)CC2CCCN(C(C3CC4C=CC3CCC4)=O)C2C1 c1(OC)cccc2c1C(C(=O)NCC1CSC1)CC2 C1(CNCC2CC(C(F)F)OC2)CC12CCCCC2 C(c1cnn(C)c1)=C(C(=O)NC1CCC(CNC(c2c(CCC)[nH]cc2)=O)C1)C c1(CNC(COCCCC#C)=O)nc(C)c(C(=O)NC2CCC(SC)C2)o1 C(CC1=CCN(C(c2c[nH]nc2C(C)C)=O)CC1)NC(C1(C)ON=C(C)C1)=O C1(C(=O)NCCCn2cc(CC=C(C)C(F)F)nn2)CC2(C1)CC(C)C2 C#Cc1ccccc1CC(N1CCC(O)CC1)=O.C12CC(C1)CC(=O)N2 C1(NC(C(CC)NC(C)=O)=O)COC2CN(C(=O)C(=Cc3ccncc3)C)CC12 C1(C(C)C)CN(C(=O)C=C2CCCC2)CCN1C(c1cccc(OCCF)c1)=O C=C(F)CN=C(NC1CCC(N2CCCC2)CC1)NC1CN(C(=O)OC)C1 NS(=O)(=O)c1ccnc(C(=O)NCC(C2CC2)NC(C2CCC(C#N)C2)=O)c1 c1(C(N(c2ccccc2)C(CC2(C=C)CCC2)=O)=O)ccccc1C.C(CO)S c1(OC)ccc(C(=O)N(C2CCCC(NC(=O)CC3CCSCC3)C2)C)c(C)c1 C(C(C)(C)CC(=O)N1CCC2(CC2C(=O)N(C2CCNC2=O)C)C1)N(C)C C(=O)(C1CCc2c[nH]nc21)NC(CCNC(C(=Cc1ccccc1)CC)=O)C C1(NC(CNC(CN2CCC(OC)C2)=O)=O)CCC(F)(F)CC1 N1(C(c2c(NC(C(C)OC)=O)cccc2F)=O)CCC2(C(=O)NC)CCCC12 CC1CC(NC(C23CC(C(F)F)(CO2)C3)=O)CN1C(=O)C=CC1CCCC1 C(CCC(=O)N1CC(C(=O)NCC(=O)N(C)CCF)C1)OC(=O)NCC N1(C(c2n(C)nnc2)=O)CC2CCC2(NC(=O)CSCc2cccnc2)C1 CC(C(=O)NC1CC(N(C(=O)CSc2ccon2)C)C1)C1CCCO1 c1(C(=O)NCC2CN(C(CCCCN(C(C)=O)C)=O)C2)cc2cc[nH]c2cn1 c1(N(C2CC3CNC2C3)C(C(C)NC(C)=O)=O)cccc(N2CCOCC2)c1 N1(C(Cc2c(C)noc2Cl)=O)C2CCC1CN(C(c1n[nH]cc1Br)=O)C2 C(=O)(C#CCOCC)NC(c1n[nH]cc1CNC(C(C)OCC=C)=O)=O.C(C)(C)(C)O c1(C(=O)NC2C(NC(c3cn(C)c(=O)cn3)=O)CCC2)c[nH]c2ccccc12 c1(C(N2CC(C)C(NC(C3CCOC3)=O)CC2)=O)cc2c(ccn2C)s1 C(CCC(O)C(=O)NCC(C)(C)CC(F)F)NC(C(C)c1cccs1)=O c1(OCC(=O)NC2CC(C)CC(C)C2)c(F)cc(F)cc1Br Nc1cc(F)c(C(=O)N(CCNC(c2cc3n(n2)CCO3)=O)C2CC2)cc1Cl Nc1nccnc1C(=O)NCCCCCNC(c1cncc(Br)c1)=O c1(C(=O)NCC2C(CNC(CCC=C)=O)C2)c(F)cc(C)cc1Br c1(C(N2CC3C(NC(C4C(C(=O)OC)C4)=O)(C3)C2)=O)cc(C(N)=O)cc(C)c1 C1(CCN(C(=O)CCc2cccs2)C)CCCCN1C(C1COCCN1C)=O C1(C(N2CC(C)CC(NC(C(CCC)NC(C)=O)=O)C2)=O)CC2C=CC1C21CC1 c1(OC(C(=O)N(CC(C)CNC(c2ncc[nH]2)=O)C)C)ccccc1C#N Cc1c(F)ccc(C(N2CC(C3CN(C(C4CC4[N+](=O)[O-])=O)C3)C2)=O)c1C C1(CC=C)(NC(=O)Cn2ccc(C)n2)CCCN(C(c2cnc(O)c(F)c2)=O)C1 CCC(CC(=O)N1CCN(C(c2cc(C)ncn2)=O)C(CS(C)(=O)=O)C1)C(C)C C(=O)(CCCCCCNC(=O)CNc1cccc(-c2ccsc2)c1)OC(C)(C)C CCC(O)CC(=O)NCC1CCN1Cc1ccc(-c2ccc(C)cc2)cc1 CCC(CNC(c1cccc(OC)c1)c1nnnn1C1CCCC1)(CC)CO C1(CCNC(c2cncc(OC)c2)=O)CN(C(C2C(C)C2C)=O)CCS1(=O)=O N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(=O)C(F)(F)c3ccncc3)CC2C1 C=CCC(C(=O)N(CC(C)NC(=O)CC1C=CCC1)CC)c1ccccc1 N1(C(c2cccc(C)c2O)=O)CCCC(C2CC2NC(c2nn(C)cc2Cl)=O)C1 c1(SC)c(C(F)(F)F)cnn1C1CCC(C(=O)NC23CC2CN(C(=O)CO)C3)CC1 c1(C(C(=O)N)N(CCOCCN(CC)CC)C)nc(O)n[nH]1.C1(C(C)C)CCCC1 C(C(CC(=O)N(C)Cc1cn[nH]c1)NC(=O)CN1CCCCC1)OC CC1CCCn2ncc(C(N3CC(O)(C(C)NC(=O)CCc4ncc[nH]4)C3)=O)c21 C1(F)(C(=O)NCC(CN(C(=O)C(c2ccc(Cl)cc2)(C)O)C)O)C(C)(C)C1(C)C C(CCC)(C(=O)N(C)CC1(NC(=O)CC(C)c2cnn(C)c2)CC1)=CCC N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3COCCO3)=O)CC2)C1 c1(C(=O)NC2CCN(C(COCCCC)=O)C(C)C2)cccc2cccnc12 Cc1nc(NC(=O)NCCC2CCCC2(C)C)nn1-c1nc[nH]n1 C1(C(=O)NC23CC(C2)C3)(CC)CCCN(C(=O)CC2CCCOC2)C1 C(CN=C(NCC(C)Oc1ccccc1)NC1CC1C)c1scc(C)n1 C(=O)(CCCCCc1cccc(O)c1)NC1C(CNC(C(=C(C)C2CC2)F)=O)C1 c1(CC(=O)O)cc2c(cc1C)OCO2.CCC(C)(CNC(c1csnc1OC)=O)O C(C)(C)(CCCNC(=O)C(c1cccc(F)c1)C)NC(C1(CC=C)COC1)=O C(=O)(CC(F)(F)C(F)F)N(CCCNC(=O)CCC(F)(F)F)CC c1(OC)cccc(C(=O)N(CC(C)C(=O)N(C)C(c2nc(C)no2)C)C)c1 C(=O)(C1=CC2(CCOC2)C1)N1CC2(OCC(C(NOCCOC)=O)C2)C1 c1(CCC(=O)NCC2CN(C(CSC)=O)C3C2C3)c(C)nc(O)nc1O C1(CCNC(=O)CCOC2(O)COC2)CCCN(C(=O)Cn2cnnc2)C1 c1(CN(CCN(C(CC2ON=C(CC)C2)=O)C)C)ccnc2ccccc12 CCC(CC(=O)N1CCC(C(=O)NCC(F)C(C)(C)O)(CC)C1)CC(C)C C1(NC(c2nsc(C)c2N)=O)COCCN(C(=O)CN(C2CCCC2)C)C1 N1(C(C2CC(C#C)(O)C2)=O)CCC(NC(=O)CNC(=O)CC)C(O)C1 Cc1sc(Cl)cc1C(C(=O)NCCCOCC1CC1)N(CC(C)C#N)C c1(CC)ccc(O)c(C(=O)N(C)CC2CCCN(C(=O)C(=O)NCC(F)F)C2)c1 c1(OC)cc(-c2cn(C(C)C(=O)N3CCC(SC)C3)nn2)ccc1O c1(C(=O)NC2(CC(=O)Nc3ccc(Cl)nc3Cl)CCC2)ccc(F)c(Br)c1 C1(NC(c2c(C)oc(Cl)n2)=O)CCN(C(=O)CCC(C)(C)C)C(C2CC2)C1 C(=O)(CCC(F)(F)C(F)(F)F)NCC1N(C(=O)C(O)CC2CC2)CCN(C)C1 N1(C(c2nnc(C)s2)=O)C2CCC1CC(CNC(=O)Cc1nccs1)C2 C1(N(C(c2cn(CC)nn2)=O)CC)CCCN(C(=O)CCN(CC(F)(F)F)C)C1 C=CCCC(C(=O)NC1CCOC1)NC(=O)CC1(C)CC1 N1(C(COC(C)C)=O)CC(C)CN(C(c2ccc(F)cc2Cl)=O)C(C)C1 C1(C(N2CC(F)(CNC(c3cc(CCCO)on3)=O)C2)=O)CN2CCC1CC2 C(=O)(CCCCC(C)C)N1CC(NC(c2ccc(C)cc2Cl)=O)C(C)C1 C1(N(C(=O)CCC(N)=O)C)CC2CCC(C1)N2C(=O)CCC1CCCO1 CC(C)CC(C)(C)NC(=O)C=CC(C)NC(C1CCCCO1)=O Cc1ccncc1-n1cc(C2(O)CN(C(C3CCC(C(F)F)CC3)=O)C2)nn1 C1(NC(C(C2CCN(C(=O)C3=CCCOC3)CC2)C)=O)CC2(CCCO2)C1 c1(C(N(CCNC(C2(C)C=CCC2)=O)C2CC2)=O)cccc2nc(O)oc12 C1(OC)CC(CNC(C2(OC)CC2)=O)N(C(=O)CCc2ccncc2Br)C1 C1(O)(CCNC(CSCC#C)=O)CCCN(C(c2nocc2C(C)C)=O)C1 c1(NC(C)=O)ccc(C(=O)NCC(C)NC(C2CN(C(N)=O)C2)=O)cc1.C(C)(C)(C)N C1(CNC(C=CCOCCOC)=O)(OC)CCCN(C(=O)CCCCCSC)C1 Cc1cc(C)c(C(N2CCC3CC23C(=O)NCc2ncnn2C(C)C)=O)cn1 c1(C(=O)NCC2(COC)CCCN2C(=O)CNS(N)(=O)=O)ccc(F)c(O)c1 c1(C(=O)NC2CC3(CNC(=O)OC(C)(C)C)C2C3)cc(O)nn1-c1nc[nH]n1 C1(C#CC(=O)N2CCC(CO)C(NC(c3ccc(F)c(Cl)c3)=O)C2)(CC)COC1 c1(C(N2CCCN(C(c3n(CC)ncn3)=O)C(C)C2)=O)ccc2nc(O)oc2c1 c1(CC(=O)NCCCCNC(=O)CC2CC3COCC23)c(F)c(F)cc(F)c1F N1(C(=O)NC(C)C=CCCc2ccccc2)CC2(CCCO2)C1 N1(C(CC2(C)CCC(=O)C2)=O)CCCC(O)(c2cn(C3CCOC3)nn2)CC1 Cc1ccc2c(C(=O)NC3CN(C(=O)CC4CCOC4)CC3C)cnn2c1C c1(C(=O)NC2CN(C(C3(O)CCOC3)=O)C2)ccn2c1CSCC2 c1(C(N(CC(=O)NC(c2cn(CC)nc2)C)C(C)C)=O)ccncc1Cl C(CC(=O)N1CC(CC(C)NC(=O)CC2(OC)CCC2)C1)OCC#C n1(CC)nc(C)c(NC(=O)C(N)CC2CC(F)(F)C2)c1C(F)(F)F C1(CC(N)=O)(CNC(C2COCOC2)=O)CN(C(C2C=CCC2)=O)C1 N(C(=NCCC1(C(F)(F)F)CCOCC1)NC(C)C1CC1)C1C(C)C1C C1(C(=O)NC2CC(OC)C2)CC(C)N1C(=O)Cc1cnn(C(C)C)c1 C(=O)(CCCCCn1cc(-c2cccnc2N)nn1)C(=O)Cc1ccccc1 N1(C(C(C2CCC2)OCC)=O)CCCCC1CCCNC(=O)CCc1cnc[nH]1 C1(C(C)NC(=O)C2=CCC2)CN(C(c2cc(C3CC3)on2)=O)CCO1 c1(C(N2CC(C(=O)NC(C3CCC3)C)C2)=O)cc(I)ccc1Cl C(=O)(C(F)CC(C)(C)NC(c1cn(C)c(C)n1)=O)NC(CC=C)CC C(CC(C(=O)Nc1cccc(Cl)c1)NC(c1n[nH]c(C)c1Cl)=O)=CC c1(CN2C(C)(C(=O)Nc3ncc(Br)nc3I)CC2)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NCC2C3CN(C(C4C(C#N)C4)=O)CC32)ccc2nc(O)oc2c1 c1(C2C(C)CCO2)c(Oc2cccc(Cl)c2)ccc2cccnc12 c1(C(N(C)CCNc2nccc(CO)n2)=O)ccc(C(=O)OC)c(F)c1 c1(CC)c(C(N2CCCC2C(C)(C)C(=O)NCC(C)O)=O)nnn1C CCCC(C(=O)N1CCOCC1)NC(C1CN(C2CCC2)C1)=O C1(C(N2C(CCNC(c3ccc(C)s3)=O)CCC2)=O)CCc2n[nH]cc2C1C Cc1cccc(C(=O)Nc2ccsc2C(N2CCOCC2C(C)C)=O)c1C Cc1ccc(Br)c(C(c2nnnn2C2CCCCC2)NCc2cncnc2)c1 C(=O)(C#CC(C)(C)O)NC(C(C)NC(c1cn(C(C)C)nc1)=O)C(C)C c1(C(N2CCC(OC)(CNC(C3CCCC3(C)C)=O)C2)=O)coc2c1CCCC2 N1(C(c2cnc(=N)[nH]c2)=O)CCC2(CC1)CCN(C(c1cccnc1Cl)=O)C2 c1(-c2nc(-c3cccc(Cl)c3)nn2Cc2ccccc2F)ccc(F)c(F)c1 CCC(CC)C(C)C(=O)NCC(C1CCCC1)NC(c1cc2c([nH]1)CCC2)=O N1(C(c2cccc(CCC)c2)=O)CCN(C(=O)C(F)CC2CCCC2)CC(O)C1 C(=O)(C(CN(C)C)NC(=O)C(C1CCOCC1)O)N(C)Cc1cn(C2CC2)nn1 c1(C(=O)NCCN(C(CC(COC)C)=O)C2CC2)cc(Br)ccc1OC N1(C(=O)OC(C)(C)C)CCC(F)(CNC(C2CC(CCO)C2)=O)C1 N1(C(c2ccn(C)n2)=O)CCn2c(CNC(C3(C)CCCNC3=O)=O)nnc2C1 c1(C(=O)NC(C(C)NC(Cc2cc(OC)nn2C)=O)CO)ccc(CO)c(F)c1 CC1CN(C(=O)CCOC2CC2)CC1CNC(c1csc(C(N)=O)n1)=O n1(CC)c(SCCCCN(C)C)nnc1-c1cc(Br)no1 N1(C(COCCC)=O)CCC2(CC1)CC(C)N(C(C1CC3C=CC1CC3)=O)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CCN(C(c2c(OC)c(Cl)ccc2)=O)C1)C c1(C(=O)NCC=CCNC(CC2C(C)C(=O)CC2)=O)cncc2c(O)nccc12 CN1C(=O)CC(CNCC2CCC2C(=O)O)C1c1ccc(Cl)c(Cl)c1 CC1(C)CN(C(=O)COCC2CC2)CCC1NC(C1(F)CCOCC1)=O N1(C(c2ccc(OCC)cc2)=O)CC2(CCC2NC(=O)CC2C(=O)NN=C2C)C1 c1(C(N2CC(CNC(CCC(C)SC)=O)C(C)C2)=O)ccc(CN(C)C)c(F)c1 C#CCCCC(C)C(=O)NC(CCC1CCC1)C(=O)NCC(C#N)CC c1(COC(C=C(CCN(C)C)Cl)=O)c(Br)ncn1C CC(CC(=O)NC1CN2CCC1CC2)C(C)(C)NC(C1C=CC=CC=C1)=O Cc1cc(C(N2CC(CNC(c3ccco3)=O)C3CC23)=O)c(C)n1C Cn1ccc2cc(C(N3CCCC3CNCC3COC4(CO)CC3C4)=O)ccc12 c1(C(N2C(CNC(CC(n3c(CC)ncc3)C)=O)CCC2)=O)nn(C)cc1N N1(C(C(C=C)OC)=O)CC2(CC(NC(C3CC34CCCCCC4)=O)CO2)C1 Cc1ccc2c(c1)C(C(=O)N1CC(NC(c3cnc(OC(C)C)o3)=O)C1)C2 C1(NC(c2ccc(CC)cc2)=O)CN(C(c2cc3ccoc3s2)=O)CC(F)(F)C1 c1(C(C)N(C(=O)C(=O)N(CCCC(O)CO)C)C)cccc(F)c1 C1(NC(C2OCCN(C)C2)=O)CN(C(=O)COC2CCC2)CCC1O C1(CC)C(C(N2CCN(C)C(C)C2)=O)CCCN1C(=O)CCOCC1CCC1 c1(OCC)ccc(C(=O)NCC2CCC(C)CN2C(=O)C2=COCC2)cc1N C1(C(=O)NCC(CC(C)C)C)CCN(C(C2CC(F)CN2C)=O)CC1C C(=O)(C(C)(O)C(F)(F)F)N1CC2C(CNC(c3ccc(C(C)C)nc3)=O)(C2)C1 CC(C)CCCCC(=O)NC1(C(=O)NC2CCC3CCC2C3)CSC1 C1(C)(C(N(CC(C)NC(c2csc(C3CCCC3)n2)=O)C)=O)CC2(CCC2)C1 N1(C(c2cncc(CC)c2)=O)CCC2(CCC2NC(=O)Cn2nnc(C)n2)CC1 c1(N2CCN(Cc3cc(O)cc(O)c3)C3C2C3)ncnc2[nH]ccc12 C#Cc1cc(F)c(C(=O)NC(CO)C(C)NC(=O)C(C(C)C)NC(N)=O)c(F)c1 C(=O)(C(C(C)C)N(CC(=O)NCC1(C)CCCC1)CCOC)OC N1(C(Cc2c(C)ccs2)=O)CCCN(C(C23C4CC(CC24)C3(F)F)=O)C(C)C1 C(=O)(C(CCCCN1CC(NC(=O)Nc2nc(Br)cs2)C1)NC)OC(C)(C)C.SC c1(C(=O)NCC2(CNC(c3c(CC)ncs3)=O)CCC2)cc([N+](=O)[O-])ccc1C c1(C(=O)NC(C2CCN(C(C3OCCC(C)C3)=O)CC2)CO)coc2c1COC2 C12(C(N(CCC)CCNC(C3CCCN3C(=O)C3CC3)=O)=O)CCCC1CCC2 C1(CNC(c2nocc2C)=O)C(C)CCCN1C(C(c1cccc(C)c1)C)=O N1(C(C(C2CC2)NC(C(C)=C2CC2)=O)=O)CCC2(C1)CN(C)C2 C1(C2CCC2)(C(N2CC(O)(C(C)NC(C3(c4ccno4)CC3)=O)C2)=O)CC1(F)F c1(OC)ccc(Cl)c(CC(=O)NCC(C2CCC2)NC(C2CC2F)=O)c1 Cc1cccc(C(=O)O)c1.C(C)(C(=O)N(C)C)N(C(CN(C(=O)O)CCC1CC1)=O)C C(=O)(C1=NOC(C)C1C)N1C(CC)C(NC(c2ccnn2C(C)C)=O)CC1 c1(OC)cnc(Cl)nc1C(N1CCC(NC(=O)COC(C)C)C1C1CCC1)=O C1(C(=O)NC(C(=O)NCCOC(C)=O)c2ccoc2)CCC(C)=C(C)C1 C#CC(C)(C)C(=O)NC(C)C(C)NC(c1c(Cl)noc1C)=O c1(COC)cc(=NCCC2C(C)CCCN2C(c2cn(C(C)C)nn2)=O)[nH]cn1 C#CCC(O)C(=O)NC1CC1CNC(c1csc(-c2ccc(Cl)cc2)n1)=O CCC1=C(C(=O)NC2CCC(C(=O)NCC3CC(C)=NO3)C2)CCCO1 c1(-c2cn(CC(CNC(c3c[nH]nc3F)=O)OC)nn2)c(N(C)C)cnn1C C#Cc1cc(NC(=O)C(=O)NCc2ccc(O)nn2)cc(F)c1 Nc1ccc(Cl)nc1C(=O)NCCCCCCNC(C1CC(=C(F)F)C1)=O C1(CNC(CCSCC)=O)CCC(C(N2CCC(CC(=O)NC)CC2)=O)CC1 N1(C(C2CC(OCC)C2)=O)CCC=C(C(=O)N2CCCC(C)(COC)C2)C1 C1(C(=O)NCCCC(C)NC(=O)CCCCO)CC(=O)NC1(C)C N12CCC(CC1)C2CC.C1(NC(C2CCOC2)=O)CCN(Cc2ccncc2)CC1 C1(NCc2c(OC(CC)C)ccc(C)c2)Cc2n[nH]cc2C(N)C1 C1(CCCCC)CCC(N=c2nc(O)c3c(ncn3C)[nH]2)CC1 CC1CN(C(=O)C(F)C(C)(C)O)CCCN1C(c1cc(Cl)ncc1N)=O CCCC(C)CC(=O)NCC(C1CCCCC1)CNC(C12CC(C1)C(C)O2)=O N1(C(C(C2CC2)OCC)=O)CC2(CCC2NC(c2ccc(OC)s2)=O)C1 c1(OC)cncc(C(N2CC=CC2CNC(=O)CCOCC(F)(F)F)=O)c1 S(=O)(=O)(c1cccc2c1OCCCO2)NC(c1ccc(=NC)[nH]c1)=O CCCC(C)C(C)(c1nnnn1CCOCC1(C)CC1)NCC(F)(F)C(F)F Cn1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCC2)=O)CO)n(C)c1=O c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)cc(S(N)(=O)=O)co1 c1(C(=O)Nc2nccs2)n[nH]c2cccc(-c3ccc(CO)cc3F)c12 N1(C(c2c(C3(C)CC3)cccc2)=O)CCN(C(C23CCCC(C2)OC3)=O)C(CO)C1 CC1=NOC2(C1)CC(C(=O)NC1(CCNC(=O)CC(Cl)Cl)CCC1)C2 c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2CCCC2)ccc(COC)s1 C1(NC(CCOC)=O)CCCC1NC(=O)COCC1CCC1 Cc1cc(C)c(CC(=O)NC2CCC(C)N(C(=O)COCC(C)(C)C)C2)c(O)n1 c1(C(N2CCC(CC(=O)NCC3(SC)CC3)C2)=O)c(C)nsc1C CCC(CN(C)C)C(=O)NC1CCCC1CC(=O)NC1CC(C(C)(C)O)C1 CC(C)(CO)CC(O)CC(CNC1CC1)CC1CCC1 Cc1cc(CC(=O)N(C2CCCN(C(=O)C(N3CCSCC3)C)C2)C)n(C)n1 Cc1cc(=NC(C)CC(N)=O)[nH]c(NC2CCc3ncccc3C2)n1 N12CCN(CC(C)(C)C1)C(=O)C(C)SNc1c(nc(C)cc1)C2=O.C(C)(C)SC CC(C)C(C(=O)NCC(c1ccc(F)cc1)C)N1CCCC1=O N1(C(Cn2c(C)ncc2)=O)CC(C)N(C(c2ns[nH]c2=O)=O)CC1C N1(C(C=CCCC)=O)CCN(C(=O)CCN(C(=O)C(CCOC)OCC)CC)CC1 c1(C(=O)NC2CN(C(=O)CN(CCO)CCO)CC2F)cc(F)ccc1Br CC1(CNC(=O)CCN2CCOCC2)CCN(C(c2cnc(C3CC3)s2)=O)C1 c1(CNC(C)=O)cccc(C(=O)NC)c1.C1(CC(=O)NCC(CO)NC)CC=CCC1 C1(NC(c2cc[nH]c2)=O)CN(C(c2coc(Cl)n2)=O)CC1n1ccnn1 N1(C(c2ccc(C(C)=O)o2)=O)CC(NC(=O)C(C#N)CC2CC2)CC1C C(N=c1nc(N2CCC(O)CC2)c2sccc2[nH]1)c1ccc(NC2CCC2)cc1 C(CC(=O)NCC1(C)CCN(C(c2ccc(CO)cc2)=O)C1)(C(C)C)OCC C1(N(C(C(C(C)C)F)=O)C)CN(C(c2n[nH]c(O)n2)=O)CC1(C)C N1(C(CCc2cc(C)on2)=O)CCC(C)(CNC(=O)Cc2ccc(Br)cn2)C1 n1(CCC)ncc(C(=O)NCC2CN(C(c3cc(F)cs3)=O)C2)c1C C(=O)(C1=NN(C)C(=O)CC1)N1C(CC)C(NC(c2cncn(C)c2=O)=O)CCC1 c1(C(N(CCOCCO)CC)=O)cn(CCNC(c2cnns2)=O)cn1 c1(C(C)C)ccc(NC(c2nc(C(N3CCCC(C)(F)C3)=O)cs2)=O)c(C#N)c1 N1(C(c2c(N)cnc(Cl)c2)=O)CC2CCCN(C(c3cnn[nH]3)=O)C2C1 C1(CC(=O)NCC2=C(C)CCC2)N(C(C2CCN(C)C2C)=O)CCC1(C)C C1(C(=O)NN2CCC(C(=O)NC3CCCC3CF)CC2)CCS(=O)CC1 N1(C(=O)NC(C2C(c3ccc(C#N)c(Cl)c3)C2)C)CCN2CCCC2C1 CC(Cc1ccccc1)C(=O)NCC(F)CNC(C1CN(S(C)(=O)=O)C1)=O c1(C(=O)NC(C2CCN(C(c3c(C)ccc(O)c3)=O)C2)C)c[nH]c2cccnc12 CC(F)(F)C(C)(C)CNC(=O)CCC1CCCN(C(c2n[nH]c(O)n2)=O)C1 CCCC(CCC)=CC(=O)N(CCNC(=O)Cn1nccn1)CC CC1(C)CCCN(S(=O)(=O)N2CCC(CF)CC2)CC1 CC1CCC(CNC(c2ccc(SC(F)F)cc2)=O)N(C(c2cnc(O)s2)=O)C1 C1(C(C)NC(=O)CCn2cc(CCN3CCCC3=O)nn2)(OC)CCOC1 O=C(C#CC1CCCO1)NCC1CN(C(=O)C2=CCCS2)CC12CCC2 CON(CCC(=O)NC(c1ccoc1)C)C(=O)C1=C(C)CCCC1 C(=O)(C(CC1CCOCC1)NC(=O)CC1CC1CC)N(CC=C)CC1CCCC1 C(=O)(CC(C(F)(F)F)NC(c1csc(O)n1)=O)N(CCOC)CCO N1(C(c2cc(Cl)ncc2Cl)=O)CCCC2C1CCN2c1ncnc2cc(Br)sc12 C1(CCC)CN(C(C2CC(F)(F)CS2)=O)CCN1C(=O)CC12CCC(CC1)C2 C1(NC(CSCCCC)=O)CCC12CN(C(c1ccco1)=O)C2 c1(NC(C2CC(C)(C(=O)OC(C)(C)C)C2)=O)ccc2c(c1)C(O)CC2 c1(NC(C(CCC#C)NC(=O)Cc2nc(=N)[nH][nH]2)=O)cccc2c1CCO2 N1(C(c2ccc(F)cc2Cl)c2nn[nH]n2)C2CCCC1CC(O)C2 c1(C(=O)NC2CC(O)CN(C(=O)Cc3ccccc3F)C2)cnc2[nH]ccc2n1 Cc1cc2ncn(CC(=O)NCCNC(=O)C=Cc3ccc(Cl)cc3)c2cc1C N1(C(c2c(C(C)C)nns2)=O)CC2CCC1CN2C(c1cnc2ncccn12)=O C1(C(=O)NC(CC#C)CC#C)CCN(C(=O)C(CC(=C)C)OC)C12CCC2 N1(C(c2cc(CNC(CCC(=O)NCC)=O)oc2)=O)CCC(CO)C(C)C1 N1(C(C2CCN(C(=O)CC3CC4C=CC3C4)CC2O)=O)CCC12CCCOCC2 C#CC1CCN(C(=O)C(F)C2CC(NC(C3(N(C)C)CC3)=O)C2)C1 C(=O)(C(CCF)NC(C1C=CCN(C(c2oc(C)cc2C)=O)C1)=O)OC C(=O)(CC(C)C(C)C(C)C)NCC1C(O)CCN(C(c2c(C)cccc2O)=O)C1 c1(C(=O)NCC(C)NC(C(C2CC2)OC)=O)c(C)cncc1F C1(CNC(C23CCC2CC3)=O)CC(F)(CNC(c2ccncc2)=O)C1 c1(OC)ccc(C)c(NC(c2cc(NC(=O)C#CC(=O)O)cn2C)=O)c1 C(=O)(C1=CNC2=NCCCN12)N1CC(CN(C(=O)C=CC=C(Cl)Cl)C)OCC1 c1(C(CSCC(=O)OC)Nc2nnnn2-c2ccccc2)cc(Br)c2c(c1)OCO2 c12cccc(c1)NC2.c1(C(N(CCN(C)C)C)=O)cccnc1N1CCCCC1 C1(O)(CNC(C=CC(C)C)=O)CCN(C(C2CCN(CC(C)C)C2)=O)C1 C1(OC)CC(NC(=O)CCc2cc(C)on2)CN(C(C2CC(C)(O)C2)=O)C1 N1(C(C(C(C)C)SCC)=O)CCOC2(CCC(N=c3nc[nH]cc3C#N)CC2)C1 C(C(C(C)(C)C)NC(=O)CC(C)O)NC(C1N(CC)CCC1)=O C1(C(=O)NCC(C)=CC(=O)NCC2CCC(=O)O2)CC12CCCC2 Cc1ccc2cc(C(=O)NC(C)CNC(=O)C(=Cc3cn(C)nn3)F)[nH]c2c1 n1(CCC(=O)NC2(C)CC(NC(C(CC)(C)OC)=O)C2)ccc(O)nc1=O c1(C(N2C(CNC(C(CC3CC3)NC(C)=O)=O)CC2)=O)ccc2c(c1)CCC(=O)N2 c1(C(CNC(c2n(COC)ncc2)=O)NC(c2ccoc2)=O)ccc(Cl)nc1 C1(c2n(C)nnn2)(NC(CC2CC2)C2CC2)CC2(CCCOC2)C1 CCCCC(CC)C(=O)NCc1occc1C(=O)NCC(CC)n1cccn1 C(=O)(CC1=CCN(C(=O)C(O)c2ccco2)CC1)NC(c1ncnn1C)C N1(C(c2ccc(CC)o2)=O)CCN(C(=O)C2=C(Cl)CCOC2)CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NC(C)CN(C)C(c1cc(F)ccc1O)=O N#CC1CN(c2ncc(I)cn2)CCN1C1CCCC1 C=C1c2ccccc2C(=O)N1CC(N1CCC(C)S(=O)(=O)CC1)=O N1(C(C=CCN(C)C)=O)CCN(C2CCN(C(c3csnn3)=O)C2)CC1 CCCCCCC(C)C(=O)NCCCC1CN(C(=O)CSCCC(C)C)CCO1 C(=O)(C(F)C(C)(F)F)NCC1(COC)CCCN1C(c1cccc(CCO)c1)=O O=C(NOCC1CCCCC1)C1=CCC(NC(=O)CCc2ccccc2)C1 c1(SCC(=O)Nc2ccc(N3CCCCC3)cc2)ccc(Br)cc1 C1(NC(CC2C(NC(C(C)N3CCCC3)=O)CC2O)=O)CCC(=O)NC1C CC1CC(n2cc(C3CCCCN3C)nn2)CCN1C(c1cc(O)nc(Cl)c1)=O c1(C(N2CCC2c2cn(CCN3CCCC3)nn2)=O)cnc2c(Cl)cccn12 C1(NC(c2ccc(OCC(=O)OC)cc2)=O)CCN(C(=O)CC(C)SC)CC1F C1(CC)(NC(c2ccc(OCCF)cc2)=O)CCCN(C(=O)C(C)N(C)C)C1 CC1(C(=O)NCC2CN(C(=O)C(F)C3CCCC3)CC2O)CC(F)(F)C1 c1(CS(C)(=O)=O)cccc(C(N2CCOC(c3cccc(F)c3)C2)=O)c1 N1(C(CC(c2c(C)noc2C)C)=O)CCC(NC(C2CSC2)=O)C(C)(C)C1 N1(C(C2C(CCOC)C2)=O)CC(CNC(=O)C=Cc2cnn(C)c2C)CCC1C C1(OC)CC(C)CN(Cc2cc(C(=O)OC(=O)OC(C)(C)C)c(C)o2)C1 C1(CCN(C)C(C2(CCO)CC2)=O)CCCCN1C(=O)CCc1cccnc1Cl C1(C(C)C)CN(C(c2ncn(C)n2)=O)CCN1C(c1cc(Br)n(C)n1)=O n1(CNC(CC2CC(SC)C2)=O)nc(C(=O)N(CC(C)O)C)cc1C Cc1ccc2cc(C(N3CCN(c4cc(F)ccc4C(C)(C)C)CC3)=O)sc2c1 c1(SC)cn(C)nc1C(=O)NC1C=CC(CNC(C2CCS2(=O)=O)=O)C1 C(C1(C)CCOCC1)=CC(=O)NCC(C)N(C(C1C(C2C(C)C2)C1)=O)C C1(C(=O)NC(c2nc(C)no2)C)(CC)CCCN1C(=O)Cc1ccn(C)c1 C1(C(N(CCNC(=O)CSc2cccc(Cl)c2)CC)=O)CCCCC12CCC2 N1(C(C2(OC)CCC(C)(C)C2)=O)C2CCC1CC(C(=O)Nc1cnn(C)c1N)C2 c1(C(=O)NCC(C)N(C(C(C)OCc2ccc(C)cc2)=O)C)ccc(C)nc1N CC1=NOC(c2nc(NC(=O)COC3(c4noc(C)n4)CC3)no2)C1C N1(C(c2ncc(C)[n+]([O-])c2)=O)CC2(CCOCC2)C1c1cn(CCCO)nn1 c1(C(N(CC2CC2)CC2CC(O)C2)=O)cnccn1.O=C1CN1 c1(OC(CCc2c[nH]c(=N)s2)=O)cc(Oc2cccs2)cc(F)c1 N1(C(c2scc(C)c2)=O)CC2CCCC(NC(c3cnoc3)=O)C2C1 N1(C(CCC)=O)CCC2(CCC(NC(C3CCC(O)CN3C)=O)CC2)C1 C1(NC(CNC(C2C(C)C2)=O)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1O CC1(C2(C(=O)NCCCCC3CC3)CC2)CC1 C1(C(=O)NCCC(C)NC(=O)C(C)(C)C2CCCO2)CCC(N(C)C)CC1 n1(CCC(=O)NCC(CN(C(Cc2cc(C)n(C)n2)=O)C)O)ccc(O)nc1=O c1(N(c2ncccn2)C(C2CNC2)=O)cccc2ccoc12.CC1C(=O)N1 c1(C(N2C(CNC(CC=CC=C)=O)C(O)C(O)C2)=O)cc(=O)c2ccccc2o1 C1(NC(CC(=O)OC(C)(C)C)=O)C2CN(C(=O)C(O)CC3CCCCC3)CC12 c1(CC)nc(CNC(c2cc(C)on2)c2nnnn2C(C)C(=O)OC)co1 C1(NC(COC)C(=O)OC(C)C)CCC2(CC1)CC(NC(C)=O)C2 C=CCC(C)(C)CC(=O)NC1COCC1NC(C1CCCN(C(=O)NC)C1)=O Cc1nn(C)c(C)c1C(C)C(=O)NCCc1cc(C(=O)O)ccc1Cl N1(CC(=O)N(C(C)(F)F)C)CCCC(NC(=O)CC2(CBr)CC2)C1 N1(C(C(C)O)=O)CC(C)N(C(=O)C=C2CCC2)CC1C C(C(=O)N1CC(C)(O)CO1)OCCN(C(=O)CC1=CCCCC1)C C1(NC(=O)C(C(=O)C(F)OC(F)(F)F)=O)CC(C#N)C1.CCCC(c1ccco1)N C(=O)(CCCS(=O)(=O)N1CC(COc2cc(C3=CC(=O)CCC3)cs2)C1)OCC N1(C(C(CC#C)NC(c2cccc(CO)c2)=O)=O)CCCC(C)(C#N)C1 Cc1ncnc2c1CC(C(=O)N(CCC(C(C)C)NC(c1ccoc1)=O)C)CC2 N1(C(C(C)NC(N)=O)=O)CCCC(C2CCCN(C(C3OCCC3(C)C)=O)C2)C1 C1(C(=O)NCCC(C)NC(CCC(C)SC)=O)Cc2c(C)cccc2N1 S(=O)(=O)(c1cccc2cnccc12)N(C(C)C(=O)N1CCCC1)CC C(CCCC(=O)NCC(C)(C)CN(C)C(C1CC(F)C1)=O)(OC)OC c1(C(N2CCCC(NC(CC3CCC(C)C3)=O)CC2)=O)c2c(nn1C)CCCC2 c1(OCCN(CCCCCC)C)cnc(SC)nc1.C1(C(N(CCO)C)=O)CCCO1 CCCC(C)(O)C(=O)NCCCC(C)NC(C12CC(C)(C1)C2)=O N1(C(CN2C(C)CCCC2)=O)CC2ON=C(CN(c3cn[nH]c3)C(=O)COC)C2C1 CCCCC(O)C(=O)NC1(C)CC(NC(=O)CC2(C)CCOCC2)C1 n1(CC(=O)NC2CC(NC(c3nc(C(F)(F)F)cs3)=O)C2)nc(O)ccc1=O C(CCS(C)(=O)=O)(C1CC1)NC(C(=O)NC(C1CC2C=CC1C2)C)=O Cc1nc(C)c(C(=O)NC(C2CCN(C(c3nnsc3N)=O)CC2)C)[nH]1 c1(C(=O)OC)ccc(C)nc1N1CCCC(CC(=O)NC2CCCOC2C)C1 c1(C(=O)NC2(C)CN(C(=O)C(F)CC3CCCC3)C2)ccc(Cl)c(S(C)(=O)=O)c1 C(=O)(C1COc2ccc(Cl)cc21)N1C(CNC(=O)Cc2nc[nH]n2)CC(O)C1 c1(C(N(C2CC(NC(CCc3cc(C)[nH]n3)=O)C2)C)=O)nccc2occc12 C12(C(=O)NCC3CCC(F)(CNC(C=C(CC)CC)=O)C3)CCCCN1CCC2 CC(C(=O)N1CCCOC(CNC(c2nscc2Br)=O)C1)C(F)(F)F C(C(=O)NNC(=O)COc1ccc(C(=O)N(C)C)cc1)C1C(C)CCO1 C1(C(=O)OCC)CN(C)C(=O)CCN(C(=O)NC2COCC2SC(C)(C)C)CC1 Cc1cc(C(=O)NC2CC(C)N(C(c3cn(-c4ccn(C)n4)cn3)=O)C2)ccn1 N1(C(CCCCCC)=O)CC2=C(C1)CN(C(C1CC(NC(=O)OC(C)(C)C)C1)=O)C2 c1(N(C(CN(CCOC)CC2CCCN2C)=O)C)ccccc1Br C(=O)(C(C)(F)C(=O)N(CC(C)NC(=O)CN1CCCC1)C)OCC N1(C(=O)NCC(C)CCc2ccco2)CCCC1CN1CCOCC1 C12(C(N3CC(C)C(CC(=O)NCC4CNC(=O)C4)C3)=O)CCCC1OCC2 C#CCC(C)(CC)C(=O)N1CCCC(C)(CNC(=O)CC2CC(F)(F)C2)C1 Cc1ccccc1COCC(=O)NC(C)C(C)NC(c1ncccc1O)=O C(=O)(C(F)(F)CCn1cccn1)NC1OCCC(NC2(C)CC=CC2)C1 CC1CC(C(=O)NCC2CC2CC(=O)NCc2ncc(CO)o2)CN1C N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(F)(F)C(O)C3CC3)CC2CC1 C1(N2CC(C(N3CC(c4cn(-c5nccs5)nn4)C3)=O)C2)CCCCC1C1CC1 Cc1ccc2cc(C(N3CCC(CN(C)C(C4CC4C(F)(F)F)=O)C3)=O)cn2c1 C1(CC(=O)NC(C(C)C)C2CCC2)CN(C(=O)COCC2CCCC2)CC1CO c1(C(N2CCC(NC(CC(C)(C)OC)=O)C2)=O)cccc(S(N)(=O)=O)c1 c1(C2C(C(=O)NC(C)CN(C(=O)CN3CCCC3)C)C2)cccnc1Cl C1(C(=O)NCCCNC(=O)Cc2cccnc2)COc2cc(F)ccc2O1 c1(C(=O)NCCCNC(c2c(CC)scc2)=O)cc(C)c(F)o1 C1(C(=O)NCc2c(C(=O)NC3COC(C(F)F)C3)c[nH]n2)CC12CCCC2 c1(NC(COC(Cn2c(C)nnn2)=O)=O)cccc(N2CCCC2)c1 c1(Cc2cn(CCOC(C(COCCOC)F)=O)nc2)cccc(S(C)(=O)=O)c1 c1(C(N2CC(CC)N(C(=O)Cn3nnc(C)n3)CC2)=O)cc2sc(C)cc2s1 C(=O)(C1CCCC1c1cccc(F)c1)OCC(C(=O)OC(C)(C)C)NS(C)(=O)=O c1(CC(N2CCCCC(NC(C3(Cl)C(C(C)=O)C3)=O)C2)=O)cnc2cccnn12 C1(CC(=O)NCC=CCNC(c2c[nH]nc2-c2ccncc2)=O)CCOCC1 c1(OCC(=O)N(C(C)CNC(c2ccc(C(C)O)cc2)=O)C)cc(F)cc(F)c1 C1(CNC(c2scc(C)c2C)=O)CCN(C(C2(C)CCC(O)CC2)=O)CC1(F)F C1(F)(COC)CCN(C(=O)C(C(=O)OC)NC(c2cccc(OCC)c2)=O)CC1 c1(NC(C23CC(C)C2C3)=O)cccc(CC(=O)NC2CC(OC)C2)n1 c1(C(=O)NCC(CCNC(=O)C=CC2CC2)O)ccn2nccc2c1 N1(C(C2C(C)CCO2)=O)Cc2n[nH]cc2C1C(=O)N1CCC2(CNC(=O)O2)C1 C12(C(=O)NCC(C3CC3)NC(C3(C)CC(C)C3)=O)CC(C)(CCO1)C2 Cc1cc(N)cnc1C(=O)NOCC(=O)N(c1cn[nH]c1)CC12CCCC1C2 C#CCCCCCCCNC(=O)C(C1CCC1)NC(=O)CC(O)CC(C)C C(=O)(CC1=CCCC1)N(C)CC1N(C(C(C2CCC2)OCC)=O)CCC1 c1(C(N(C)CC2N(C(C3(CC(C)C)CCCC3)=O)CCC2)=O)cccnc1O c1(C(C)NC(=O)NC2(N)CC2)ccc(C2CC2)c(C(F)F)c1 c1(C(N(CC(C)NC(c2cc(CO)[nH]n2)=O)C)=O)nccn2ccnc12 N1(C(c2scc(C)c2)=O)CCC2CCN(C(C3(C)CNC(=O)C3)=O)CC12 c1(OC)ccc(OC)c(C(=O)NC(C)CNC(C2CCCCS2)=O)c1N c1(N2CCC(C)(NC(=O)CC3CCCC(=O)N3)C2)ncc(C#N)cc1F CCCCCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C=CC=C(Cl)Cl)C1 C1(CC(=O)NC(c2cccc(C)c2)C)CCCN(C(=O)C=CC2(C)COC2)CC1 c1(C(=O)NC2(CNC(COC)=O)CCC2)cc2c([nH]1)CCOC2 C=CCC(CC)C(=O)NC1(c2cn(CC=CC=CC)nn2)CCOC1 N1(C(c2c(CC)c(F)ccc2)C(=O)NC(C)CC)C(C)CS(=O)(=O)CC1C CC1CCC(C(=O)N2CC(n3cc(CN(C4CC4)CC4CC4)nn3)CO2)CC1C n1(CC)nc(C)cc1C(=O)NCC1CC1c1cccs1.C12CN(C1)C(=O)C=CC2 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(O)C(F)(F)F)ccc2cc[nH]c2c1F C1(NC(c2cc(-c3csc(CO)c3)cs2)=O)CCCC12CC2 C1(NC(C2(CCC=C)CC2)=O)COCC1C(=O)NCC(C)SC C1(C(C)NC(=O)Cc2ccnn2C)CCN(C(C2CC2C2CCCO2)=O)CC1 N1(C(C2C(CC)CCC2)=O)CCCOC(CCNC(c2nnsc2C)=O)C1 CC12CCC(C)(O1)C(C(=O)NCCN(C(=O)CCCn1cncn1)C1CC1)C2 C1(C(N2C(CNC(CCC3(C)CC3)=O)CCC2)=O)C2CCC1(C)C2(C)C N1(C(CCC(C)OC)=O)CC2CC2CC(NC(c2c[nH]cc2Br)=O)CC1 C(=O)(CCCOC(C)(C)C)NCCN(C)C(c1cc(-c2ccccc2)ns1)=O N1(C(Cc2cc(C)nn2C)=O)CCC(NC(=O)CC2CC2(C)C)CC(C)(C)C1 C=C(C)C(O)CC(=O)NCC1CCC1NC(c1cc(-c2csc(C)n2)c[nH]1)=O N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(C12CCCC1C2Br)=O C(=O)(C1=CCC(F)(F)CC1)NCC1(CNC(C(C(C)SC)O)=O)CCOCC1 C1(C(=O)NC(C)CNC(c2ccc(OCC(N)=O)cc2)=O)CCc2c[nH]nc2C1 c1(NC(CCSCC)C)cc(=NC2CC3CCC(C2)O3)[nH]c(C(C)C)n1 c1(NC(C2N(Cc3ccc(OC)cc3)CCC2)=O)ccc2c(c1)C(C)(C)C(=O)N2 c1(OC)cc(C(=O)NCc2ccc(-c3ccc(NC(C)C)nc3)cc2F)cc(C)c1 Cc1ccc(Cl)c(O)c1C(=O)NCC1CCCC(CNC(=O)C2=CC(C)(C)C2)C1 c1(NC(=O)CC2CCCN2Cc2cnc(Cl)s2)ccc2cnccc2c1Cl CC1(C)CCC(F)(F)CC1C(=O)NCC=CCNC(c1cccc(N)n1)=O CS(=O)(=O)CCCCCN=c1[nH]c(=NCCn2cnnc2)c2[nH]ccc2[nH]1 CC1(C)CN(C(=O)C(C)(C)c2cccs2)CC(CNC(=O)CNC(=O)C2CC2)O1 N1(C(Cc2ccc(C)cc2)=O)CCN(C(=O)C(C)n2ccnc2)C2CC12 Cn1cc(C(=O)NCC2CC2NC(=O)C=C2CCSCC2)c(C(F)F)n1 C1(N(N2CCN(C3CN(C(=O)C#CC(=O)N(C)C)C3)CC2)C)CCn2cnnc2C1 c1(C(=O)NCCC(C)NC(C2CCC(C)CC2)=O)cc(=O)c2ccncc2o1 C(C(F)(C(=O)N1CCCC(C)(C#N)C1)C(C)C)NC(C1CC(OCC)C1)=O N1(C(CCc2n(C)c(S)nn2)=O)CC2CCN(C(C3(F)CCCCC3)=O)CC2C1 Cc1cc(=NCC2CC(NC(c3c(C)nn(C)c3C)=O)C2)[nH]c(C)n1 c1(C(=O)NC2(CCC)CC2)ccoc1CNC(=O)C(C)(C)OC CCC(C)C(=O)NCC(=O)NC1(NC(=O)CN2CCCCC2)CC(CO)C1 N1(C(C(F)=C(C)C)=O)CCCC(CCNC(c2ccnc(NC(N)=O)c2)=O)C1 O=C(C1=CC2(CCN(C(=O)CSC(F)F)C2)C1)NC1CCCCC1O C1(C(=O)NCC2CC3CN(C(C(CC=CC)C)=O)CC32)CC2(C1)CS(=O)(=O)C2 N1(C(C2(C#C)CC2)=O)CCC2CCN(C(=O)Cc3cccc([N+](=O)[O-])c3C)C2C1 C1(C(=O)NCC(C)(C2CC2)NC(c2c(CC)occ2)=O)CCN(C)C1C N1(CCCOc2c(OC)cnc(C(F)(F)F)n2)C2CCC1CN(C)C(=O)C2 C1(CC(=O)NC(C)CC(C)O)(COC)CN(C(=O)CN(C(=O)C(C)C)C)C1 c1(C(=O)NCC(C2CC2)NC(CCSC)=O)cc(C#N)c(F)cc1F CCC(C(=O)N(C1CCN(C(=O)CC2(CO)CC2)C1)CC)n1nccc1C C12C3CCC1N(C3)C(=O)N2.c1(OC)ccc(Br)c(OC)c1 C1(NC(C2C(NC(C(C(C)C)=O)=O)CCC2)=O)CCCC2(CC1)CC2 CN1C2CCC1CC(=CC(=O)NC13CCC1CN(C(c1cccc(F)c1)=O)C3)C2 c1(CNC2CCN(CC)C2=O)ccc(SCc2nc(C(C(=O)OC)C)on2)cc1 CC1CC(C(N2CCC2(C)CCO)=O)CCN1C(c1csc(F)c1)=O C(=O)(C1=CCC(C)CC1)NCC12OCC(NC(C(C)NC(=O)NC)=O)(C1)C2 N1(C(C=CC(C)(C)SC)=O)CCC2(CC1)CCN(C(=O)Cn1ccnc1C(C)C)C2 C1(C(=O)OCC)C2CN(C(C3(CC)CCC3)=O)CC12 N1(C(COC(C)(C)C)=O)CCC(NC(C2(S(N)(=O)=O)CC2)=O)C12CCC2 C1(C(=O)NC(CC)C(F)(F)F)CN(C(=O)Cn2ccnc2C)CCC1(F)F c1(N2CC(NC(C(C)OCCC(C)C)=O)(CO)C2)ncc(I)cn1 C1(C(=O)NCc2n(CC)cnn2)CCN(C(c2sccc2Cl)=O)C1C C(=O)(CCCN=[N+]=[N-])N1C(CC(=O)NC(C=C)C2CCC2)CC1 CC(C)CCC(=O)NCCCC(C)NC(c1ccc(C2CCCCC2)s1)=O c1(C(=O)NC2CC(C)(NC(C)=O)C2)cncc(O)c1Cl.c12ccc(o1)C(=O)NC2 C1(CC#C)(C(N2CC(N=[N+]=[N-])C2)=O)CCN(C(=O)CC2CCCO2)C1 N1(C(C(CC)N(C)CC)=O)CCN(CCNC(C2CC(n3cnnc3)C2)=O)CC1 C12(NC(c3scc(C(N)=O)c3)=O)CCCC1CN(C(C13CCC(CC1=O)C3)=O)C2 C(=O)(C#CC(C)(C)CNC(c1nc(O)sc1C)=O)N(CCSC)CC C1(C(=O)NC(C)C(=O)N(C23CC(C2)C3)C)CCOC1=O CC(C)C(O)CC(=O)N1CC(NC(c2ncc[nH]c2=O)=O)CC(O)C1 C(=O)(C1CSc2ccccc21)N1CCC(NC(C2NC(=O)OC2)=O)C(CO)CC1 N1(C(c2c(OC)nccc2)=O)CCC(C2CC2)C1CNC(c1ccccc1C)=O CC1CC2CN(C(=O)C(O)CC[S+](C)C)CC2N1C(C1CC(O)C1)=O c1(C(N2C(C(=O)Nc3c(OC)cc(O)cc3)C(C)CC2)=O)cc2cccn2cn1 C1(NC(=O)Cc2ccnc(O)c2)CC2CC1CN(C(C13CCC(CC1F)C3)=O)C2 N1(C(CCC(C)OC)=O)CCC2(CC1)CN(C(C1CCCC(F)(F)C1)=O)C2 c1(C(=O)NCCCCNC(C2CC2C(=O)NCCO)=O)coc(-c2cccs2)n1 c1(C(N2CCC(CCNC(c3n(CC)ccc3)=O)C2)=O)cc(C2CC2)ccc1F c1(OC)cc(C(=O)NCC2(NC(c3ncn(CC)c3)=O)CCCCC2)cc(C)c1 N1(C(c2nn(CC)c(C3CC3)c2)=O)CC2(CC2)CC1CNC(=O)CCC(F)F C1(C(=O)NC(C)CCC(F)(F)F)COCCN(C(c2cc3n(n2)CCC3)=O)C1 C1(NC(C2CCCN2CC(F)F)=O)CN(C(=O)COC2CCOCC2)CC12CC2 CC(C)C(C)CC(=O)N1CCCC1CCC1CCN(C(C2(C(F)F)CC2)=O)CC1 CC1CCN(C(=O)C(C)(C)C2CC2)CC1CNC(=O)CCC1(O)CCC1 c1(Nc2c(C(=O)OC)ccc(C)n2)ncc2c(ncn2C)n1.C12CCCC1NC2 c1(NCC(=C)Cl)cc(N2CCCC(CO)C2)nc(C(F)(F)F)n1 N1(C(C(CC=CCC)C)=O)CCC(CNC(c2nn[nH]c2Cl)=O)C12CC2 N1(C(CN(C2CC(C#N)C2)CC(=O)NC2CC=CC2)=O)CC(=O)NCC1C(N)=O c1(NC(C2N(c3ncc(C)c(C)n3)CCCC2)=O)cc(Br)c([N+](=O)[O-])cn1 C1(CC)CC(c2nnnn2C2CC(F)(F)C2)(NCCC=CBr)CCO1 C1(NC(C)=O)CC2(C1)CN(C(c1cccc(C(F)F)c1F)=O)C2 N1(C(=O)CCOc2ccc(F)cc2)CCC2CN(C(=O)C3=CCCC3)C2C1 c1(C(C(=O)N(C2CN(C(C(CC)SC)=O)C2)C)O)ccc(Br)cc1 CC(C)C1=NOC(C(N2CCCC2CNC(c2c(C3CC3)cccc2F)=O)=O)C1 N1(C(c2c(C)sc(O)n2)=O)CC(NC(C2(C)CC=CCO2)=O)CC12CCOCC2 N1(c2n(CC(C)C)c(-c3cnn4cc[nH]c34)nn2)CCCC(C2CCC2)C1 C1(C(N2C(C)CN(C)CC2)=O)CCN(C(=O)C(C)N=[N+]=[N-])CC1(C)C C(=O)(C1=CC2CC=CCC12)NCC1(CNC(c2cc(C)c(Cl)c(N)c2)=O)CCC1 C1(NC(c2scc(CC(N3CCCC3=O)(C)C)n2)=O)CC2CC1CN2.C(=O)(C1CC1)N C1(NC(c2[nH]c3ncn(C)c3c2)=O)CCN(C(c2cc(Cl)no2)=O)CC12CCC2 C1(CNC(C(c2ccc(Cl)cc2)C)=O)CN(C(=O)CC2COCCO2)CC1C c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)N(C)C)=O)cccc2c1CCN2 Cn1cc(C(F)(F)F)cc(C(=O)NCCCNC(=O)CCCCCF)c1=O C=CCCCCC(=O)N1CCOC(CNC(C2CC(Oc3ccccc3)C2)=O)C1 CC(C)(CC(F)(F)F)C(=O)NCCOC1CCN(C(=O)CN2C(=O)CCC2=O)C1 CC(CC(=O)NC1CCC1CNC(=O)C1=CCCS1)C(F)(F)F c1(C(=O)NC2CCC(C(=O)Nc3occ(C)n3)CC2)ccn2nccc2c1 C(=O)(CC(C)(C)C(F)(F)F)NC(CN(C(=O)C(c1cccc(F)c1)(C)O)CC)C CC1=C(C(=O)NCC2CC3CN(C(=O)C(C)Cc4ccnn4C)CC23)CCC1 c1(C(=O)NC(CNC(C(CCC)OC)=O)C2CC2)cc2n(n1)CCNC2=O C1(C)(C(N2C(CN(C(=O)CC3CN(C(C)=O)C3)CC)CCC2)=O)CCCNC1=O Cn1c(C(N2CCN(C3CC3NC(=O)CC(=O)N(C)C)CC2)=O)ccc1[N+](=O)[O-] c1(C2C(C(N(CCCNC(C(CC)(C)O)=O)C)=O)C2)c(Cl)cccc1Cl C(CC(C)C)(C(=O)NCC(CC(C)C)NC(c1coc(C2CCC2)n1)=O)OC C1(O)(CNC(C2(COC)CCC2)=O)CCCN(C(=O)CCn2ccc(C)n2)C1 c1(CNC(N2CC(COC)CC2(C)CO)=O)cc2ccncc2[nH]1 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CC(C)NC(=O)CCC3(C)CC3)c12 N1(C(C(C)C2CCCC2)=O)CC2(C(=O)NCCCC(C)(F)F)CC1CO2 N1(C(CC)=O)CCN(C(c2ccc(CC)nc2)=O)CC(O)C1 C(C(C)(COC)CC)NC(C(C=CC)O)=O.C1C(=O)N1CC(C)C C1(C(=O)N(CCN(CCOC)C(C2(C(C)(C)C)CCC2)=O)C(C)C)CCC(=O)N1 C(C1CCc2cc(F)ccc21)NC(=O)Nc1ccc(C(F)(F)F)cc1 C1(CCNC(CN(C)C)=O)CN(C(=O)C(CO)NC(N)=O)CCO1 N1(C(C=CC=CCC)=O)CC(CNC(c2cncc(CC)c2)=O)CC1(C)C N1(C(C(C=C=C)C)=O)CCN(C(=O)OC(C)(C)C)C(CO)C1 C(=O)(CCS(=O)(=O)c1cccc(Br)c1)NCCNC(C(C=C=C)C)=O N1(C(c2ccc(OC)s2)=O)CC=CC1(C)C(=O)NCCC1CCCC(C)C1 C(c1ccncc1)=CC(=O)NC1CC(CNC(c2nnc(C(F)(F)F)s2)=O)C1 C1(CNC(c2c(C(=O)OC)ccnc2)=O)CCN(C(=O)C=CC(=O)N(C)C)C(C)C1 N1(C(CCN(CCC)C)=O)CCC(NC(c2[nH]cnc2C)=O)C1C N1(C(CC(CC2CC2)NC(C2(CC(C)=O)CC2)=O)=O)CC2CC1CS2=O C12(CNC(Cc3cccc(OCC)c3)=O)CCCC1CCN2C(=O)CN(C)C N1(C(CCN(C(c2cc(OC)n[nH]2)=O)CCO)=O)CCC([N+](=O)[O-])CC1.C1CN1 N1(C(c2c(N)nccn2)=O)CCCC(NC(c2nn[nH]c2Cl)=O)C(F)C1 C1(CNC(CC2N(C(C)=O)CCC2)=O)CCN(Cc2cnn(C(C)C)c2)CC1 C#Cc1ccnc(C(=O)NC(C)CCN(C)C(c2cc(=O)c(Br)c[nH]2)=O)c1 c1(-c2cn(CCOCCNC(=O)COC(F)F)nn2)ccc(F)cn1 N1(C(c2cnn[nH]2)=O)CCC2CN(C(=O)Cn3ncn4nccc4c3=O)CC2C1 CCC(C)(F)C(=O)N1CCC(CNC(c2cc(CN(C)C)on2)=O)C1 CCC(CC)(C(=O)NC1CC(C)N(C(c2cccc(N)c2)=O)C1)OC N1(C(=O)NCCCOc2c(COC)cccc2F)CCC12CCCOC2 Cc1ncc(N)cc1C(=O)NC(c1cn(C)nn1)CNC(=O)Cc1ccncc1 C1(C(C)N(C2CCN(CC)C2)C)CCN(C)CC1 N1(C(C2OCCCO2)=O)CCC(C(=O)NC2CC3CCC2C3)=C(F)C1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2cnn(C3CC3)c2Cl)=O)CC1(C)C C1(CNC(CN(CCC)C)=O)CCCCCN1C(C1CC(OC(F)F)C1)=O C1(C(=O)NC(CCC)c2nn[nH]n2)CCn2c(C(F)(F)F)nnc2C1 C#Cc1ccnc(C(N2CC(NC(=O)CCc3ccc(F)cc3)CC2C)=O)c1 c1(CC(=O)N(CCCCO)C(CC(C)(C)O)C)cnc(C(F)(F)F)cc1 N1(Cc2scc(C)n2)CCOC(C)(C(N(C(C)C)CC(=O)C(C)(C)C(F)F)=O)C1 C1(NC(c2scc(C)c2)=O)CCOCC1NC(=O)C(c1ccn(C)n1)C CN=c1c(C(=O)NC(C)C(C)NC(=O)Cn2cncc2C)c[nH]c2ccccc12 C1(C(=O)NCC(CCC)OCC)C(C)OCCN1C(c1conc1CC)=O N1(C(C(C)N(CC)CC)=O)CCC2C(NC(=O)CCc3cnc[nH]3)CC12 c1(C(C)(C)NC(C2OCC(C)C2)=O)ccc(-c2cn(CC(C)(C)C#N)nn2)cc1 c1(N2C(CNC(c3c(CC)noc3)=O)CC3(CC3)C2)nc(O)c2ccccc2n1 C(c1ccc(O)cc1)=CC(=O)NCCOC1CCN(C(C2CCS2(=O)=O)=O)C1 C1(C(=O)NC(C)CC(=O)NC(C)Cc2ncn(C)n2)(OC)CCOCC1 c1(CC(=O)NCCC(CC)(C)NC(=O)C=CC(C)(C)SC)cccc(C)c1C N1(C(C(CC)OC)=O)CC2(CCCCN(C(C3(OC)CCCC3)=O)C2)C1 N1(Cc2cncc(C)c2)CCC2(CCN(c3cc(C)ncn3)C2)C1 CC(C)C(C(=O)N1CC(Nc2cc(C3CC3)ncn2)C(C)C1)c1cccnc1 C1(CCC)CN(C(C2CCC3(CC3)C2)=O)CCN1C(=O)CCCCCOC C1(C(=O)NCCCN(C(C)C)CC)CCc2nc(-c3cccc(C)c3)sc2C1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(C)cc2)O)cc(C(N)=O)ccc1C N1(C(CCCOCCC)=O)CCC(C2CC2)C1CNC(c1ccc(Cl)nc1C)=O C(=O)(C1=NN(c2ccccc2C(C)C)C(=O)C1)NC12CC(NC(CC)=O)(C1)C2 C#CCCCC(=O)N(C1CCN(C(=O)C=C2CCCO2)CC1)CCOC Cc1n[nH]c(C)c1C(C)C(=O)NC1CN(C(=O)C(c2ccccc2)C)CC1CO c1(NC(C)=O)cccc(-c2cn(CC3CCC(OC)C3)nn2)c1.C1(SC)CCCCC1O c1(CNc2c(C(=O)Nc3c(Cl)cc(C)cc3Cl)nccc2)cccc2cnccc12 C1(NC(c2n(C)nc(CC)c2Cl)=O)CC2CCC1N(C(=O)CC(C)C(C)C)C2 S(=O)(=O)(c1cc(Br)c(F)cc1F)NCC1N(C(C2C(C(=O)O)C2)=O)CCOC1 c1(C(N(CCCCNC(C(C)N(C(C)=O)C)=O)C)=O)cccc(Cl)c1O N1(CCC)C(=O)CCC1C(=O)NC(CNC(=O)COCC(=O)OC)C(C)(C)C CCCCC(CC(=O)Nc1ccc(F)c(CO)c1)NC(C12CCCN1CCC2)=O C(=O)(CCCCCNC(=O)Cc1n[nH]c(C)n1)N1C(CC)(CC)CC1 CC1C(C)N(C(c2nc3ncccn3n2)=O)CCN1C(C12COC(CF)(C1)C2)=O C(=O)(CS(=O)(=O)C(C)C)N1CCC(NC(CCn2ccc(C)n2)=O)C(F)C1 C1(C(=O)NC2(C(=O)NC(C)Cc3cn[nH]c3)CC2C)CC2CCC(C1)C2 N1(C(c2ccc(C(F)(F)F)[nH]2)=O)CCCCC2(CCN(C(=O)C(Cl)=CCl)C2)C1 c1(NC)cccc(C(N2CC=CC(NC(=O)C=C3CCC(C)CC3)C2)=O)n1 c1(N2CCC(C)C(NC(c3c(C)oc(C(C)C)n3)=O)C2C)ncc2ncn(C)c2n1 c1(CC(N2CC(NC(C=C(C)C)=O)C(C(F)(F)F)C2)=O)ccc(CO)c(C)c1 Cc1ncccc1NC(C1CN(C(C2CCNC(=O)C2)=O)CCO1)=O C1(NC(CC=CC(C)(C)C)=O)CCCC(C(=O)NCC(O)C2(Cl)CC2)C1 c1(OC)cc(O)c(C(N2CC3CC3C2)=O)cc1OC.C12CC(C1)C(=O)N2 c1(C(=O)NC(CC(=O)NC(CC(=O)NC)C2CC2)C2CC2)cncc(C)n1 C1(C2CCOCC2)(CNC(CN(CCC)C)=O)CCN(C(=O)CC2CCOC2)C1 C1(C(=O)NCCOCC(=C)C)CCC(O)CN1C(c1ccn(C)c1CC)=O N1(C(C=CC=CCC)=O)CCC(C(N2CCCCC2C(F)F)=O)(OC)C1 c1(C(=O)NCC2(F)CC(CNC(=O)Cc3cnc[nH]3)C2)cc(F)cc([N+](=O)[O-])c1 c1(OC)ccc2c(c1)CC(C(=O)Oc1cncc(-c3cccnc3)c1)O2 CCC(C)C(O)C(=O)N1CCN(C(c2ccc(C(C)(C)C)cc2)=O)C(CCO)C1 c1(C(C(F)(F)F)NC(=O)C(N2CCCC2CN2CCCC2)=O)ccc(Br)cn1 C1(NC(CSCC=C)=O)CN(C(C2CCN(CCF)CC2)=O)C(CC)(CC)C1 CC1CN(Cc2cc(Cl)cc(I)c2)C(C(F)(F)F)CO1 N1(C(=O)C=CC2CCCC2)CCC2CN(C(C3CC(=O)C34CCC4)=O)CCC2C1 C1(NC(c2c(C(C)C)ocn2)=O)CCC(O)CN(C(=O)CP(C)(C)=O)C1 C(CC(=O)N(C1CCC(NC(=O)CCCN(C)C)C1)C)(C(F)(F)F)OC N1(C(C(C)=CC)=O)CC2(CCO)CCC1CC2.c12cccc(c1)NC(=O)COC2 C1(C(=O)NC2CCN(C(c3ccn(CC)n3)=O)C2C2CC2)CS(=O)(=O)CC12CC2 C1(NC(c2cccc(CC=C)c2)=O)CC(C(=O)NC(C)CCF)=CC1O C1(CNC(C=C(COC)C)=O)CC(C)CCN1C(=O)C(C)n1cncn1 c1(N2CCC(CNC(C(C)OCCCCCC)=O)C2)cc(C)ncc1C#N N1(C(c2c(C)cnn2C)=O)CC(C)CN(C(c2cnc(C(F)(F)F)s2)=O)CC1C c1(C(=O)NCC(C)CNC(=O)CCC2CCN(C)CC2)cc(C#N)c(N)cc1O N=c1[nH]c(=NCCn2ccnc2)[nH]c(=NC(CF)c2ccccc2Br)[nH]1 Cc1cc(N)c(C(N2CCCCC2CCNC(C2(C)CCCO2)=O)=O)cc1C c1(CC(=O)NCC(C)(O)CNC(c2cnoc2C2CC2)=O)cnc(O)nc1O CC1(C)CN(C(C2CC3(C2)CC(F)C3)=O)CC(CNC(c2cncs2)=O)O1 C1(NC(CN(C2CCCN(C(C3N(CC)CCC3)=O)C2)C)=O)CCCCC1(C)C C1(C(C)NC(c2cocn2)=O)CN(C(c2cnc(Cl)cn2)=O)CCO1 C1(C)(CNC(C(CCOC)(C)C)=O)COCCN(C(C2CC(C)C2)=O)C1 N1(C(c2n[nH]c(C)c2O)=O)CCOCC(NC(=O)CN(C2CCC2)C)C1 N1(C(C2(F)CCN(C(Cn3c(C)cc(C)n3)=O)CC2)=O)CCCC12CCOC2=O c1(C(=O)OC(C)(C)C)ccc(C(=O)NCC2(NC(c3cnc(S)[nH]3)=O)CC2)o1 C1(C(=O)NCC2(O)CN(C(c3nn(C)c(F)c3)=O)C2)CC2OC(=O)OC2C1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCC(CNC(C(C)OCC)=O)C1(C)C C1(CC(=O)NC(C(=O)NC(C=C)(C)CC)CSCC)CCCC12CC2 C=CC(CC)CC(=O)N(C)CC1(O)CCN(C(c2cnc(OC)c(C)c2)=O)C1 N1(C(CC2CN(C(c3cc(CCC)[nH]n3)=O)C2)=O)C(C)CCCC1C C1(C2CCN(C(=O)CNC(=O)NC3CC3)C2)(NC(=O)CC2COC(=O)C2)CC1 c1(C(=O)NC(C2CCCN2C(=O)C2=NNC(=O)CC2)(C)C)cnn2ccccc12 C=CCC(C)(C(=O)N1CC(C)(C)CC1CNC(c1ccncn1)=O)N(C)C C1(=CC(=O)NCCC2COCCN2C(c2ncccc2F)=O)CN2CCC1CC2 c1(Cn2cc(C3CCCN(C(=O)CCCCCF)C3)nn2)ccc2scnc2c1 C1(CC(C)C)C(=O)NC(C)C(=O)NO1.c1(C2(COC)CC2)cccnc1 c1(CCC(COC(CC=CC)=O)C)cccc(C)c1 C(=O)(CCCCC(C)C)N1C(CCCNC(CCSCCC)=O)CCC1 C1(CNC(C(C)CO)=O)CCC2CN(C(c3coc(O)n3)=O)CCC2C1 N1(C(C2CC(N(C)C)C2)=O)CCC2(CCC(NC(C3CSCC(=O)N3)=O)C2)CC1 C(=O)(CCCS(N)(=O)=O)NC1CCN(C(C(c2ccc(C)nc2)(F)F)=O)CC1C N1(C(c2nnc(C)s2)C)CCC(C)(NC(=O)CC2CC=CC2)C1 Cc1cc(NC(=O)C(C)(C)C2CCN(C(=O)C(C)O)C2)cnc1O N1(C(C2N(c3ccnc(NC)n3)CCC2O)=O)CCCC2(CCCNC2=O)C1 Cc1ccc2[nH]c(C(=O)Nc3ccc4c(C)nn(C)c4c3)c(Cl)c2c1 Cc1cc(=O)oc2ccc(OCC(=O)NCC(O)CCNC(=O)CN(C)C)cc12 c1(CC(=O)OC(C2COCC2O)=O)csc(N(c2ccccc2)C2CCCC2)n1 Cc1cc(=NCc2nc3ccccc3o2)[nH]c(N2CCCC(O)CC2)n1 C1(C(N(CCCNC(CCC=C(C)C)=O)C2CC2)=O)CC1C1CCCC1 c1(C(=O)NC2C(NC(=O)CCc3ccon3)CC2)ccccc1OC(F)F c1(C(=O)NCCC(O)C(=O)N2CC(N3CC(F)C3)C2)ccn2nccc2c1 N1(C(C(C2(C)CC2)OC)=O)CCCC1C(=O)N(C1CCN(CC2CC2)C1)C c1(OC)c(C(N2CCCCC2c2ccccc2Cl)C(=O)NCCSC)cccc1F N1(C(CN(CC)CC)=O)CC(NC(c2cccc(-c3nccs3)c2)=O)CCC1C N1(C(COCP(C)(C)=O)=O)CCC(NC(=O)CC2CC2C(F)(F)F)C(O)C1 Cc1c(C(=O)NCC2N(C(c3ccc[nH]3)=O)CCC2(C)C)c[nH]c1C#N c1(C(=O)NC2(C(=O)NC3(N4CCCC4)CCSC3)CC2)ccccc1Cl C1(NCC(=O)NCC(C)(C)Sc2cccc(Cl)c2)CC1C1CCCC1 C1(N(C(C(C)OCC=C)=O)C)CCCN(C(=O)CSCCC(C)C)CC1 c1(C(N2CC(O)(NC(C3CC(C(=O)OC)C3)=O)C2)=O)cnn(CC2CCC2)c1C C1(OC)CN(C(=O)Cc2ccns2)CCC1NC(=O)CN1CC2CC2C1 S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CCN(C(c2c(N)c(F)c(Br)cc2)=O)CC1 n1(CC(=O)NCC(CC)NC(c2csc(C)n2)=O)nnc(=O)[nH]1 C1(CC(N2C(CNC(COCCCC#C)=O)CCC2)=O)(C(=O)OC)CCOCC1 c1(C(C(=O)NCCOC)N(CC=C)CC#N)cccc(C2CCCC2)c1 c12cc(nc(C(C)C)n1)N2.C1(CC)CCC(C(N2CCN(CCF)CC2)=O)CC1 C1(C(N2C(CCC)CCC2)=O)N(C(=O)CC2CSC2)CC12CCCC2 C1(C(=O)NC(c2ccc(F)cc2)CNC(CCCNC(N)=O)=O)CCCC1(C)C N1(C(COC(C)=O)=O)CC(C(=O)NCc2cncnc2C)C2(CCC2)C1 CCCCC(CCC)NC(=O)CC(C)(C)NC(C1CC(F)C(=O)N1)=O C12(CNC(CC)=O)CCCCC1N(c1ncc(I)cn1)CC2 N1(C(=O)C=CCN2CCOCC2)CCC2CC(C1)CN(C(=O)C(O)C1CCCC1)C2 c1(C(=O)NC2CC(NC(C3(F)CC(C(=O)OCC)C3)=O)C2)c(CC)cccc1Cl C(C(C)(C)C(=O)N(C1CC(C(=O)Nc2cnc(SC)nc2)C1)C)SC CC1(C)CC(CC(=O)NCCC2CCCC23CC3)CN1C(=O)Cn1cnc(=N)[nH]1 c1(C(=O)NCC#CCNC(=O)C(F)(F)c2nccs2)ccc(NC2COC2)cc1 Cc1cc(C(N2CCCC(O)(CN(C(=O)CN3CC=CC3)C)C2)=O)c(C)cn1 c1(C(=O)NCCC2(OC)CN(C(C3(C)CCCS3)=O)C2)cnn(C)c1C(F)F c1(NC(CCn2cc(C3(C)CCCO3)nn2)=O)ccc(Br)cc1F C1(NC(CCC)=O)CCCCCC1NC(=O)CCC(C)(C)c1ccccc1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(=O)Cn2cc(C#N)cn2)CCC1C Cc1c(C(=O)NC2CC(NC(C3CC4CC4C3)=O)CC2O)ncn1C C12(NC(=O)Cn3cc(C(F)(F)F)cn3)CC1CN(C(c1ccc(CO)cc1)=O)C2 Cc1cnc(NC(CC2CC2)CO)c(S(=O)(=O)NCc2ccnc(Cl)c2F)c1 c1(C(N2CCN(C(c3c(SC)cn(C)n3)=O)C(C)C2)=O)ccc2c(c1)OCO2 C1(NC(C23CC(CNC(=O)OC(C)(C)C)(C2)C3)=O)CC1C1CCOCC1 Cc1nc2sccn2c1C(=O)N(C)CCN(C(=O)CO)C.c1(OCCF)cnn(C)c1 c1(C(N(CCCN(C(c2cccc(OC)c2N)=O)C)C)=O)cc(S(N)(=O)=O)co1 N1(C(C(C2CC2)NC(Cc2nc(C)oc2)=O)=O)CCC(C(C)C)(CO)C1 N1(C(C(OC)OCC)=O)CCC(N(C(=O)CN(C)C(c2cccs2)=O)C)C(C)C1 N1(C(C(=O)NCC(=C)C)C2CC(C(=O)OC(C)(C)C)C2)CCCC1CC C1(C(=O)NCCCCC)CCCCCC1n1cc(C(C)(O)CC)nn1 c1(OC)c[nH]c(C(=O)NCCC(Cc2ccccc2)NC(C2(Cl)CC2)=O)cc1=O C1(c2cn(CC3(O)CCN(C(CC)=O)C3)nn2)CC2(C1)OCCO2 C(=O)(C1=NOCC1)N1C(CN(C(C2(c3ccc(F)cc3)CCCC2)=O)CC)CCC1 c1(C(=O)Nc2nsc3ncccc23)cc([N+](=O)[O-])c(O)cc1F.CC12CN(C1)C2 C1(NC(Cc2c(C)n[nH]c2)=O)CCN(C(=O)C(C)(C)N2CCOCC2)CC1F c1(C(=O)NCC(C2N(C(C(CC#C)C)=O)CCC2)(C)C)ccc(OC)c(C)c1 Cc1onc(C(N2CCC23CN(C(C2CCC(=O)N2C)=O)C3)=O)c1[N+](=O)[O-] C1(CNC(CCCOC)=O)CN(C(c2ccc(C(=O)NC(C)C)[nH]2)=O)CCO1 c1(OC)cc(F)ccc1C(=O)NC1(CNC(=O)C(C)CC2CCC2)CC1 N1(C(C(C)NC(Cc2nc(C)oc2)=O)=O)CC(C)(C)OCC1C N1(C2CN(C(C(COC)O)=O)C2)CCN(C(=O)C=CC(C)(C)C)CC1 N1(C(COCCC=C)=O)C2CCC1CC(CNC(c1cccc(OCC)n1)=O)C2 c1(CC)cn2c(n1)CCC(C(=O)NCC1C=CCN1C(c1cnsc1)=O)C2 N1(C(CCCC)=O)CC2CCC(C1)N2C(=O)Nc1c(Cl)cc(Cl)cc1Cl c1(NC(C2(NC)CCC2)=O)cc2c(F)c(F)cc(F)c2[nH]1 c1(C(=O)NCC2OCC(CNC(=O)CC3OCCO3)C2)ccc2ncnn2c1 c1(C(N2CC(CNC(C=CC=CC)=O)C2)=O)cnc(S)n1-c1ccc(Br)cc1 c1(C(=O)NC(CCNC(C(C(C)C)C)=O)C)cc(Cl)cc2c1CCC2 C1(C(=O)NC2CN(C(c3cnc(SC)n3C)=O)C2)CCN2CCOCC12 c1(C(=O)NCC(C2CCN(C(=O)CO)CC2)(C)O)ccccc1[N+](=O)[O-] c1(CC(=O)NCC(C)NC(=O)CCN2CCOC2=O)cccc(N2CCCC2)c1 C1(NC(c2cc(CC)c(=O)n(C)c2)=O)CC12CCN(C(c1nn[nH]c1Cl)=O)CC2 N1(CC=C)CCCN(C(=O)C(C2CCC2)NC(=O)CC2COCCO2)CC1 c1(N2CCCC(CN(C)C)C2)nc(N2CCCOC(C(C)C)C2)c2ccsc2n1 C1(C(=O)NC(C=C)(C)CC)CCN(C(=O)Cc2cccs2)C1(C)C C1(NC(CCC2N(C)CCC2)=O)CN(C(=O)CC2CCCOCC2)CC2(CC2)C1 C1(C(=O)NC2CN(C(c3c(OC)csc3)=O)C(C)(C)C2)CC(C)(C)OC1(C)C c1(SC)cccc(C(=O)NC2CCCC2NC(=O)C2=CCOCC2)c1[N+](=O)[O-] c1(OC(C)C)ccc(NC(c2c(Br)ncn2C)=O)cc1Br N1(Cc2cc(Cl)cc(I)n2)CCC2CCCC(C2)C1 N1(C(CC(C=C)CC)=O)CCc2c(cnn(C)c2=O)C1 C(=O)(C1=CCC(NC(=O)C(C)CC(N)=O)C1)NC1(COC)CCCC1 N#Cc1cc(C(N2CC(CCn3cc(C4CCCOC4)nn3)C2)=O)ccc1F CS(C)(=O)=NCC(=O)N1CCC(n2cc(-c3cnn(CCF)c3)nn2)C(F)C1 CC1(C)CC(NC(c2cc[nH]n2)=O)CN1C(c1cc(C2CC2)nnc1O)=O c1(SCC)ccccc1C(=O)NCC1CN(C(c2sc(CO)nc2C)=O)C2CC12 c1(C(C)(F)F)ccccc1C(N1CCN(C(=O)CC2CCC3CC23)CC1)=O N1(C(CCC(C)C)=O)C2CC1CN(C(=O)CNC(=O)COc1ccccc1)C2 N1(C(C(CCC)OC)=O)CCN(C(=O)COc2ccon2)CC(O)C1 N1(C(C(C(C)C)n2cnnc2)=O)CCC(C)N(C(C2CC(C)(C(=O)O)C2)=O)CC1 CCCCC(C)C(=O)N(C(C)CNC(=O)CC(C)N(C)C)C c1(CC)nc(C(F)F)oc1C.C1(=O)NCCC2(CC2)N1 N1(C(C2C(CCOC)C2)=O)CCCC(C)(C)C1C(=O)NC1CC(C)CCC1O C(=O)(C(C)SC(F)(F)F)NC1(CNC(COC)=O)CC1 N1(C(CC2(C)CCOCC2)=O)CCC2(CC1)CC2CNC(=O)C(F)(F)C(F)(F)F c1(C(=O)NCC2(CNC(CCN(C)CC)=O)CCCC2)cccc(C(C)C)c1N O(NC(=O)C(C)(C)CCNC(=O)C(C)CC(=O)OC)CCC S(=O)(=O)(c1ccc(NCCCC2CCOC2)cc1Cl)N1CCC(CC)(CO)C1 CC1(NC(c2ccccc2)=O)CCN(C(=O)CC2CCCC(C#N)C2)CC1 N1(C(C(=O)NCCc2cc(F)ccc2F)=O)CCc2c(Br)cc(F)cc2C1 C1(CNC(C=COCC)=O)CC2(CCOCC2)CN1C(c1cc(O)n(CC)n1)=O C(=O)(C(CC(C)C)ONC(C1CC(=O)NC1(C)C)=O)NC(CCC)CO c1(CC)nnc(C)cc1C(=O)N(C(c1ccccc1)CNC(C1CCSC1)=O)C c1(CC)ccc(O)c(C(=O)NCC2CN(C(C3CCCC3O)=O)CC23CC3)c1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)C(O)CCC(C)C)CCC12CCC2 CCC(N)CCC(=O)N1CCCC(C(=O)NCc2occc2C)C1 Cc1cc(C)c(C(=O)NCC(C)CNC(c2cn(C(C)(C)C)nc2C)=O)[nH]1 C(=O)(C(C)CC(F)(F)F)N1CCC(C#C)(C(=O)Nc2ccccc2OC)C1 C1(O)(CN(C(CCCSC)=O)C)CCN(C(c2cnoc2-c2ccoc2)=O)CC1 C1(CN(C(=O)COCCCF)C)CN(C(=O)CC2CCCS2(=O)=O)CCO1 C(=O)(C1NCc2nc(C)ncc21)NCc1ccc(C)c(F)c1F C12(NC(C(c3ccc(F)c(F)c3)(C)C)=O)CCCC1CN(C(c1ccsc1)=O)C2 C1(C(=O)NC(CCC)C(=O)NCCOCCCO)CCCCC1(C)C CN1CCCC(C(C)(C)C(N2CCC(F)(CNC(c3cc(CO)cs3)=O)C2)=O)C1 c1(OC)ccc(C)nc1C(=O)NC1(CO)CN(C(c2cc(CO)[nH]n2)=O)C1 N1(C(c2ncc(OC)cn2)C(=O)Nc2ccccc2)CCC(C)(O)CC1 Cc1nc2sccn2c1C(N1CCC(CNC(=O)CC(O)C(C)C)C12CCC2)=O C1(NC(c2cc[nH]c2)=O)CCCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 C1(NC(c2nc(-c3cccnc3)cs2)=O)CCNCC1CO N1(C(CC(CNC(C2CC(OC)C2)=O)OC)=O)CC2CC(O)CC1C2.C1(C)CC1 c1(CNC(C2C3CN(c4c(OC)c(C)ncn4)CC32)=O)ccc2oc(C)nc2c1 CC(CC(=O)N(C1CCC(NC(=O)CCC2(C)CC2)CC1)C)C(F)(F)F N1(C(CC=CC)=O)CCC2(CO)CN(C(=O)CCSc3ccc(O)cc3)CC2C1 c1(CC(=O)NC(C)C(=O)NC2CCCC(C)(C)C2)ccc(F)c(F)c1 c1(C(=O)NCCC2CN(C(C#CC(C)C)=O)CC2C)noc2c1COCC2 C1(C#N)(C(=O)NCC(CNC(CC(C)OC)=O)OC)CC(=O)C1 c1(N2C(CC#N)CN(Cc3cc(I)ccc3O)CC2)ncc2cc(Br)cnc2n1 C(=O)(C1=CC2CCCC12)NCC1(CNC(c2[nH]c(=NC)sc2)=O)CC1 Cc1ccc(C(=O)NC2(CO)CN(C(c3cc(C(F)F)nn3C)=O)C2)nc1C CCCC(C(O)C(=O)NCC(C)(C)CO)NC(C1(C)CCOCC1)=O N1(C(c2nc(NCC#C)oc2)=O)CCC(c2n[nH]c(C3CC3)n2)CC1 C(C(C)(C)CC(=O)O)NC(c1cnn(C(C)C)c1N)=O C12(NC(c3ccnnc3O)=O)CCCC1N(C(=O)C=CBr)CCC2 C(=O)(C1=CS(=O)(=O)CCC1)N1C2CC(NC(=O)C=CCN3CCCC3)CC1CC2 N1(C(C2ON=C(C)C2)=O)CCC(N=c2ccn3ccnc3[nH]2)CC1C N1(C(C(C2CC2)OC)=O)CCC2(CCCC2NC(=O)CC2CCCC3CC23)CC1 C1(C(C)C)N(C(C2C3CCCC23)=O)CC12CCN(C(=O)C(=O)NC(=O)C1CC1)CC2 C1(C(=O)NC2CCN(C(C(CN(C)C)O)=O)CC2)Cc2nccn2C1 CC(C(=O)NC(C)(C)CN(C)C(c1ccc(C2CCC2)nc1)=O)C(F)(F)C(F)F CN1C(=O)C(=O)N(CC(=O)NCc2ccnc(N3CCNCC3)n2)C1=O C1(C(=O)NC2CCSCC2)(CNC(C(C)C2CCCC2)=O)CC2(CC2)C1 N1(Cc2c(C)ccs2)C(C(=O)Nc2ccnc(C(N)=O)c2)CCC1C c1(OC)ccnc(C(N2CC(CCNC(c3conc3C3CC3)=O)C2)=O)c1C C(CCCCCNC(=O)CC1CCCC1NC(=O)C(O)C1CCC1)OC c1(OCC(=O)NC2C(NC(C(C)O)=O)CCCCC2)cccc2cccnc12 C1(CNC(CC(C)OC)=O)CC2(CO1)CN(C(=O)C(C)(F)c1ccccc1)C2 Nc1nc2c(cc1C(N1CC3CCC(C1)N3C(C1CCCCO1)=O)=O)CCCC2 N1(C(c2[nH]cc(OC)c(=O)c2)=O)CCC2CCCN(C(C3C4CCCC34)=O)C2C1 N1(C(COCCCCC)=O)CCC(N(CCC)C(C2(C)CCOC2C)=O)CC1 c1(C(CO)N)c[nH]c2ccccc12.C1(NC(C2CCN2C2CC2)=O)(CO)CCC1 Cc1ccc(O)c(C(N2CCC(NC(=O)Cc3ccco3)CC2)=O)c1 C1(CN(C)C(C2CCCN2C(=O)Cc2cncs2)=O)CCCC2CC12 C(C(C)(C)Cc1ccccc1)NC(=O)NCC=CCNC(COC)=O N1(C(CC2C(CNC(C3CN(C(C)=O)C3)=O)C2)=O)CCOCC(C)(C)C1 C(C(C)(C)CNC(=O)CC1CC1(Cl)Cl)N(C(=O)Cn1ccc(C(F)F)n1)C NS(=O)(=O)c1c[nH]c(C(=O)NCC2CCCC(NC(C3(C(N)=O)CC3)=O)C2)c1 c1(NCCN(C(c2cc(CC)ncn2)=O)C)nc2c(cc1C#N)CCC2 N1(C(c2cc(OC)nn2C)=O)CC(C2(NC(=O)Cn3cc(C(C)O)nn3)CC2)C1 c1(CC)c(C(=O)N(C)CC2CCCC2NC(C2CSCCS2)=O)ccn1C CC1CCC(CCNC(C2(CNC(=O)C(N)=O)CC3(CC3)C2)=O)CC1 N1(C(C(CC)C(F)(F)F)=O)CCC(C2(NC(c3nc(=N)cc[nH]3)=O)CC2)CC1 c1(OC)cc(OC)c(C(=O)NCCCNC(=O)C(C2CCCO2)OC)c(OC)c1 N#CC1(O)CC(C(=O)NC2CCCN(C(=O)Cc3cscn3)C2)C1 C1(C(=O)NC(C)=O)CC2(CC2)C1.C12(C)CC1NC2=O.C12CN(C1)C(=O)CO2 CCCCC(CNC(C1CC1C)=O)NC(c1ccoc1C(C)C)=O Cc1c(C(=O)NCC(C)CN(C(=O)CC(C)C(F)F)C)cc(C(C)C)n1C c1(C(=O)NCCS(C)(=O)=O)cc(=NCc2ccc(I)cc2F)cc[nH]1 N1(C(C2(C(N)=O)CC2)=O)CC(N(C(=O)COCC2CCC2)CCO)C1 Cc1onc(Br)c1C(=O)N(CCC(C)NC(C1CC1F)=O)C N1(C(c2c(CC)nns2)=O)CCCN(C(c2ccc(C)cc2)=O)C(CO)C1 N1(CCOC)CC2CC1CN2C(=O)CC1CC1CNC(=O)Cc1ccco1 C(C(=O)NC(CC1CCC1)CO)(N(C(=O)CSC(F)F)C)C1CC1 N#Cc1ccc(C(F)(F)F)nc1N1CC2CC1C2C(=O)Nc1csc(Br)c1 C(=O)(C#CC1CCCCO1)NCC1C(NC(c2ncc(C)cc2F)=O)CCC1 C(=O)(C(O)C(C)(C)C)NCC(C)N(C(=O)COc1cccc(Br)c1Cl)C CC(C)(O)C#CC(=O)NC(CNC(=O)C(C)(C)CC1CCCC1)CO N1(C(c2c(C)cn(C(C)C)c2)=O)CCCC(C)C1CNC(=O)CC1CC(C2CC2)C1 C1(CC)(NC(=O)Cn2ncnn2)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 C1(NC(C(C)N(C(C)=O)C)=O)CC=C(C(=O)NCC2CCCCCCC2)C1 CC(C)C(C(=O)NOCC(F)(F)F)N(C(=O)CCCCC1CC1)C N1(C(c2n(OC)cnc2C)=O)CCC2(CC1)CN(C(=O)CC1(OC)CC1)CCO2 CC1(C)CN(C(=O)C=Cc2cc[nH]n2)C(CNC(=O)CSC(C)(C)C)CO1 C1(NCC(C(=O)OC)c2ccsc2)CCCNS1(=O)=O N#Cc1cc(Br)ccc1C(=O)NC1CCN(C(C23CCCC2C3)=O)C1 C(=O)(CC(C)(C)CC(=O)N1CCC2C1CCCN2C(=O)Cn1ccnc1C)OC N1(C(COC)=O)CCC2CCN(C(n3c(-c4ccccc4)c(C)sc3=O)=O)C2C1 n1(C(C)C)ncc2c(N3CC=CC3)[nH]c(=NCCc3ccc(C4CC4)cc3)nc12 C(N=c1[nH]c(=NC2CC2C)[nH]c2c1CSC2)c1ccc(OCC(C)C)cc1 c1(CC)nc(C)c(C(=O)NC2CCC(N(C)C(c3ccncc3C)=O)C2)s1 N1(C(C(C)Cn2cccn2)=O)C2CCC1CN(C(=O)COc1ccsn1)C2 CS(=O)C=CC(=O)NC1CN(C(C2CC3CCC2O3)=O)C1 C1(N(C)C(c2cnsc2)=O)CCN(C(=O)C=CC(c2ccccc2)=O)CC1 CC(C)(C)C(C(=O)N1CCCC1)Oc1ccncc1-n1cc(-c2cc[nH]n2)nn1 C(=O)(C(C)(F)C(C)(C)F)N1CCN(C(C=C(CCC)C)=O)C(CC(C)(C)C)C1 C1(C(N2CCC(C)(NC(=O)C(=O)N=S(C)(C)=O)C2)=O)CCCN(S(N)(=O)=O)C1 c1(CN2CCC(O)(C(=O)Nc3ccc(SC)nc3)C2)ccn(C)c(=O)c1 O=C(O)C(Cc1ccsc1)C(=O)N1CCCC1c1ccccc1Cl.C1(S)CCCC1 CC1CN(C(=O)CSC(C)(C)C)CC1n1cc(C2C(Cc3cccs3)C2)nn1 n1(CCCCCNC(C)CC2CCS(=O)(=O)C2)c(=O)oc2ccccc12 C1(CCNC(C=C(CC)C)=O)CN(C(c2ncn(C(C)C)n2)=O)CCS1(=O)=O C1(C(N(CC(CC)NC(c2cncc(N)c2)=O)C)=O)CCS(=O)(=O)C1(C)C c1(C(N(CC(C)NC(=O)C(C)(c2ccccc2)N(C)C)C)=O)cncn1C C(C)(CCCC(=O)N(C(C)C(C)C)C1CC1)NC(c1ccc(OC)nc1)=O CC1C(NC(=O)C(C)(C)CC(F)F)C2CCN1CC2 N1(C(C2C(CCOC)C2)=O)CC(CCNC(=O)CC2CN(C)C2)C(C)C1 C1(NC(c2c(C)cc(C)[nH]2)=O)CN(C(=O)C(C)C2CCC2)CCC12CCOCC2 O=C(Cc1cc(F)ccc1C(=O)O)N1CC2COCC2O1 CC(C)C(C#N)C(=O)NC1C=CC(CC(=O)NC2CC(CCN(C)C)C2)C1 C(=O)(C(C)C(C)C(C)(C)C)N(CCOC)CCNC(c1cccnc1CO)=O CCC(C)C(C)C(=O)N1CCC(C)(CCNC(c2cc(Cl)ccc2N)=O)CC1 C1(N)CC2CC(C1)N(C(=O)C(C)=C(C)C)C2.CCCCCC=CCC=O c1(C2C(C(=O)NCC(C)N(C(c3cccc(N)n3)=O)CC)C2)ccc(F)c(F)c1 CCC(CCC(C)C)NCCOc1ccc(F)c(Cl)c1 Cc1ccc(OCC(=O)NCC23COC(CNC(c4cnco4)=O)(C2)C3)cc1 O=C(C1CCCc2nnnn21)NC1CCOCC1NC(C1(C2CC2)CC1)=O C(=O)(C(C(C)(C)C)SC)N1C(C)(CC(=O)Nc2cc(COC)oc2C)CC1 C(CC(C)C(=O)N1CCCC1(C)CCC(=O)NCC1(C)CCCC1)=CC CN1C(=O)CC(C(=O)NC(CC2CCCC2)CO)C1c1ccc(Cl)cc1 c1(CNC(C(C2CN(C(=O)CCc3cc(C)[nH]n3)C2)OC)=O)ccc(C(N)=O)s1 c1(C(N(C2CCN(C(c3cccc(CO)n3)=O)C2)C)=O)ccc(C#N)c(Cl)c1 C1(C)(C(=O)NC2(CCCNC(c3c(OC)ncc(Cl)c3)=O)CC2)CCCNC1=O C1C(C(C)C(C)C)NC(=O)CC1.c1(C(=O)N)cccnn1.CCS(=O)(=O)N C1(CC(C)C)COCCN1C(=O)C(=O)NC1(CO)CC1(C)C C1(NC(c2c(C)cco2)=O)CCCCC1NC(=O)C(C)(c1ccccc1)N(C)C c1(CN)ncc(C)cc1O.c12ccc(cc1)CC2NC(CCC#C)=O.C(C)(C)(C)O CC1(C)CC(C(=O)Nc2cnc(Cl)c(F)c2)CN(CC(N)=O)C1 C1(CNC(c2c[nH]nc2Cl)=O)CC2(CC2)CN1C(C1CC2CC2C1)=O CCC(CNC(c1ccsn1)=O)(CC)NC(C1CCN(C2CCOC2)CC1)=O C1(F)(CNC(C(c2ccccc2)OC)=O)CCN(C(=O)C(C)(F)F)CC1 CCC(CC(=O)N1CCC1Cn1cc(C2CC23CC3)nn1)C(F)F N1(C(CCC)=O)CCC(CCNC(=O)C(O)c2ccco2)C1 C1(CCNC(=O)OC)CCOC(C)C1.C1C(=O)NOCC(=O)N1C C=CCC(C(=O)NC1CCC(NC(=O)C(CO)NC(=O)C(F)(F)F)C1)C(C)C C(=O)(C#CC(C)(C)C)N(C)CC1CCN(C(c2cncc(NC)n2)=O)C1 Cc1cc(=NCC(C)NC2CC(=O)N(C3CC3)C2)[nH]c(N(C)C(C)C)n1 C(C)(C)(C(=O)NCCN(C(c1cn(CCF)nn1)=O)CC1CC1)OCCC Nc1c(C(N2CC3CC(NC(=O)Cc4cnc(C5CC5)[nH]4)C2C3)=O)ccnc1F C1(OC)CC(CNC(=O)C(C(C)C)c2cc(C)no2)N(C(=O)CCF)C1 c1(NC(CCCCn2cc(C(COC)(C)O)nn2)=O)ccc(S(C)(=O)=O)c(C)c1 c1(C(=O)NCC(CC(C)C)NC(c2cccc(O)n2)=O)coc2c1C(=O)NCC2 N1(C(C(C2CCN(C(=O)C(F)OC(F)(F)F)C2)C)=O)CC(O)C(O)C1CO C1(NC(C2CCN(C)C2)=O)C2CC1N(C(=O)CC1CCCN1C(=O)C1CC1)C2 C(C(=O)NCCC1CCN(C(=O)C(C2(O)CCCC2)F)C1)(C(C)C)NC(C)=O N1(C(=O)C(F)n2ccnc2)CCOCC(CNC(C2CC(OC3CC3)C2)=O)C1 CCC(CO)C(=O)NCCCCC(C)NC(c1scnc1C)=O C1(NC(CC(CC)C)=O)CN(C(=O)Cc2ccc(F)cc2Cl)CC2(CCC2)C1 C1(CCOC)CN(C(c2sc(=N)[nH]c2C)=O)CCN1C(c1ccn(C)n1)=O C(CCF)(C(=O)NCCNC(=O)C(C)C)NC(c1c(CC)c[nH]c1)=O N1(C(C(CCC2CC2)NC(CCc2n(C)cnc2)=O)=O)CCC12CCC(O)CC2 N1(C(C2C(=C)C2)=O)CCCC(C2(NC(C3CC(O)C3)=O)CC2)C1 N1(C(C=CC2(C)COC2)=O)CCC2(CC1)CC(NC(=O)CCCC(F)(F)F)C2 C(=O)(CCCCC(F)F)N1CCC(N(C(=O)COCC2CCCCO2)CCC)C1 CCC(CC)CC(=O)NCC=CC(N1CC=CC1(C)CO)=O N1(C(C(c2ccccc2)C)=O)CC2CCC1CN2C(c1c[nH]ccc1=O)=O N1(C(c2cc(SC)oc2)=O)CCOC2CN(C(=O)Cn3cncn3)CC12 C1(C(=O)NCCOCCO)CC2(CCN1C(C1CNC(=O)O1)=O)CC2 C(=O)(CC(C=C)CC)N1CCC(N(CC#C)C(C2CCCC2C)=O)CC1 c1(CN=C(NC(C=C)C)NC2CC2C2CC2)cc(OCC)c(O)cc1C O=C(C1=NOC2(CCN(Cc3cc(Br)cc(Br)c3)C2)C1)NCc1cc(Br)co1 CN1CCc2cc(C(=O)NCC34CCC3CCN4C(C3CCCC3)=O)ccc21 C(=O)(C#CC1CCOC1)NCC(c1ccc(C)cc1)NC(C1CC(O)C1)=O N1(C(c2nc(C(C)OC)sc2)=O)CCC(O)(C2CCN(C(=O)C=CCO)CC2)C1 C12(NC(C3(C=C)CCC3)=O)COC(CNC(=O)CC(n3nc(C)cc3C)C)(C1)C2 c1(C(N2CC3(C2)CN(C(c2csc(-c4ncc[nH]4)n2)=O)C3)=O)ncc(Cl)cc1Cl C1(CNC(C=CC)=O)CC(NC(c2c(N)c(C(F)(F)F)nn2CC)=O)C12CCC2 c1(C(N2CCCC(C)(CNC(C(C)C3CC3)=O)C2)=O)cc(C#N)ccc1F c1(CC(=O)N(CCCNC(C2CC2C)=O)CC)noc2ccc(OC)cc12 c1(C(C)(C)C)ccc(O)c(C(=O)NCC=CC=CCNC2CC(n3cnnc3)C2)c1 C(c1c(Cl)cccc1Cl)=CC(=O)NC1C(F)CCN(C(COCCSC)=O)C1 c1(OC)cc(C(=O)NCC2CCCN2C(=O)CC23COC(C)(C2)C3)ccn1 C(C)(C)(CN1C(=O)C(=O)c2ccccc21)C1(C(N2C(CC)CCC2C)=O)CC1 C(=O)(C(C)C(CC)CC)NCC1C2CN(C(C(CC(=C)C)OC)=O)C1C2 c1(NCC2C(C(=O)Nc3cc(N4CCNCC4)ccn3)C2)ccc(Br)c(C#N)c1 N1(C(C2CC(N(C)CC)C2)=O)CCCC(CCNC(=O)CCF)C1 N1(C(C(CC)OC)=O)C2CCC1C(NC(c1cccc(N(C(C)C)CC)c1)=O)C2 c1(C(CSC)NC(C2CC2F)=O)ccc(CC(=O)NC2CC(CCC)C2)cc1 N1(C(C2C(CCOC)C2)=O)CCCC1C=CC(=O)NC(C(C)C)C1CCCC1 C(=O)(C1c2cnn(C)c2CCN1C(=O)OC(C)(C)C)N(C)CCc1c[nH]c(=N)s1 c1(SC)nc(N(C)Cc2ccccn2)cc(N2CCC(NCC(C)C)CC2)n1 C1(CNS(N)(=O)=O)CCSC12CN(C(C13CCC(n4cc(SC)nn4)(CC1)C3)=O)C2 C(CN=c1[nH]c(C#N)c(Cl)s1)(C(C)(C)C)NC(C1Cc2c(cn(C)n2)CC1)=O c1(C(=O)NCCOC2CCN(C(c3c(C)coc3C)=O)C2)cc2n(n1)CC(F)C2 n1(CC(=O)NCC)cc(CNC(=O)CN(C(=O)C(CC)OC)C2CC2)nn1 c1(C(N(CC(C)N(C(=O)CC(=O)c2cnn(C)c2)C)C)=O)ccc(O)cn1 N1(C(c2cc(CC)no2)=O)CCSCC1CCNC(=O)CC1OCCC1C CN1CC(NC(C2(NC(c3ccncn3)=O)CC2(C)C)=O)C(=O)N1 C1(CC=C)(NC(=O)C(F)(F)c2nccs2)CN(C(=O)C(c2cncnc2)C)C1 C1(C2CCN(C(=O)CC3C=CCCC3)C2)CCCCN1C(=O)C(F)CC1CC1 Cc1cc(C(=O)NC2CCCC(NC(=O)Cc3ccc(F)c(F)c3)C2)cc(C)c1 C1(NC(CSc2nc(C)[nH]n2)=O)CCCCC1NC(=O)C(C)NC(N)=O c1(C(N(C2CC(NC(=O)CC3CCCOCC3)C2)C)=O)cc2cccnc2[nH]1 Cc1cc(Cl)cc(C(=O)NCCN2CCN(C(c3cc(=O)cc[nH]3)=O)CC2)c1O CC(=O)CCCC(=O)NC1CC(F)CN(C(=O)CCN2CCN(C)CC2)C1 N1(C(CNC(CCC)=O)=O)CCC(O)(C(N2CCC(C)(CO)CC2)=O)CC1 CCC(CC)C(C)C(=O)N1CC(O)CC1CNC(=O)C(C)=CC(C)(C)C N1(C(C2N(C(C3CCN(OC)CC3)=O)CC(O)C2)=O)CC2CCCC2C12CC2 N1(C(C(F)=C(C)C)=O)C(C(=O)NC2(n3ccnn3)CC2)CC1C C1(CNC(c2ccc(C)cn2)=O)CCC(C)CN1C(c1nscc1Br)=O N1(C(c2nn[nH]c2Cl)=O)CC(NC(C2(CO)CCC2)=O)CC2(CCOCC2)C1 c1(C(=O)NCC2CN(C(c3cccc(OCC(C)C)c3)=O)C2)nnn2c1CCC2 CCC(N=c1nc2c(ncn2C)c(N(CC(C)(C)CSC)C)[nH]1)c1ccncc1 c1(SC)nccc(N(C(=O)COC(C2COCC(C)O2)=O)C2CC2)n1 N1(C(C(C)S(C)(=O)=O)=O)CC2CCN(C(=O)C(C)(Cl)Cl)CC(C2)C1 C1(NC(CCOC)=O)CCN(C(c2ccon2)=O)CC1c1ccccc1 N1(C(CCOCCCOC)=O)CCC(C)(C)C(NC(c2ccc[nH]2)=O)C1 N1(C(C(C)NC(c2cc(Cl)ccc2Cl)=O)=O)CCNCC2(C)CCCC12 C1(CN(C(=O)CCOC2COC2)C)CCCCN1C(=O)C(F)(F)c1ccsc1Cl C1(CCNC(C(=Cc2ccncc2)C)=O)CCN(C(=O)CSCC#N)C(C)C1 CCCCCC(O)C(=O)NC12CC(C(=O)NC3CCCC4(C3)N=N4)(C1)C2 CC(CCNC(=O)C(C)NC=O)N(C(=O)CSCc1ccco1)C C1(C)(COC)CN(CC(C2CCC(F)(F)CC2)C)CCO1 c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)O)cc2c(o1)CCCNC2=O c1(Oc2ccc(C(=O)NC(C3CCOCC3)CC)cc2)ccc(Br)cc1Cl n1(CCN(CC)CC)cc(C2CC(NC(c3csnc3Cl)=O)C2)nn1 c1(C(=O)NCCN(C(C(CC)F)=O)CCOCCO)oc(C)nc1C Cc1cc(N)ccc1C(=O)NCC(C)(C)CN(C)C(C1CCN1C)=O c1(C(N2CC(CCNC(=O)C(O)Cn3cncn3)(OC)C2)=O)cncc(N)n1 C12(NC(c3cc(C)cc(C)c3)=O)CCCC1N(C(=O)CC1CCCCO1)CCC2 C(=O)(C(C)C(O)CC)NCCCC(C)(C)NC(c1c(CCC)nco1)=O C(=O)(C(C)CC(C)(C)C)NCCC(C)(C)NC(CSc1ccc(C)cc1)=O N1(CC(=O)NC2CCC(NC(C3C(C)OCC3)=O)C2)CCS(=O)CC1 CC(N=c1ccnc(NCc2cccc(Cl)c2F)[nH]1)c1cccc(C#N)n1 Cc1nc(C2CCCN(C(C3C4CN(C(=O)CC5CC5)CC34)=O)C2)oc1C(=O)O CC(CC(=O)OC(C)(C)C)NC(C1CSCN1C(=O)CCCC1CCCC1)=O C1(CCNC(c2c(CC)nn[nH]2)=O)CCCN(C(C2CC(C#N)(OC)C2)=O)C1 N1(C(c2ccn(C)n2)=O)CCC(C2CCCN2C(C2CCC(=O)N2)=O)CC1 C1(C(N2CC3CCCC3(CNC(=O)C(F)(F)C3CC3)C2)=O)Cc2ccccc2C1 CC1CC(NC(c2cccc(Cl)n2)=O)CCN1C(=O)C=CS(C)=O C1(C(C)C)(C(=O)NC2CCCC2C(=O)N(C)Cc2ccco2)CCCC1 N1(C(CC(CC)C2CC2)=O)CC2CN(c3ncnc(O)c3Br)CC2C1 N1(C(C)C)CCN(C(=O)NCC(C2CCOCC2)F)CC1C C1(CC(=O)N(CCCOCCN(C)C(c2cccs2)=O)C)CCCCC12CC2 N1(C(c2c[nH]c(=N)s2)=O)CC2(CCCCN(C(c3cc4ncccc4s3)=O)C2)C1 C(=O)(C(=O)N=c1nc(-c2cnn(C)c2)[nH]s1)N(CC(c1ccccc1)CO)C C1(CN(C(=O)CCC2CCCO2)C)CCCCN1C(c1ncoc1Br)=O C1(c2nc(CNC(CSC)=O)[nH]n2)CCCN(C(C2CCCCN2C(C)=O)=O)C1 C1(CC)C(=O)NCCCN1C(=O)C(CNC(=O)COCC(C)(C)C)CC1CCCC1 c1(C2c3cn(nn3)CCC(=O)N2)cc(P(C)(C)=O)cs1.CC(=O)OC1CC1 c1(CC(=O)NCC(CNC(C2CCN(CC)CC2)=O)O)nsc2ccccc12 N1(C(CN(CCC(O)C(F)(F)F)C)=O)CCC2(CC1)CC2C(=O)NC1CCC1 c1(C(N2C3CN(C(C(CC)N(C)C)=O)C(C3)C2)=O)cc(Cl)cc(F)c1F N(C(=NCCOC)NCc1cnn(C)c1)Cc1nc(CC)sc1 c1(OCC)ccn2c(C(=O)NC3CCN(C(=O)CC(C)CF)C3)cnc2c1 c1(OCC)cncc(C(=O)NCC(C)NC(c2ccc(CF)cc2)=O)c1 N1(C(COCC(C)C)=O)CCCCC(N(C)C(C2CN(C(C)C)C2)=O)C1 C1(NC(c2cnc(C3CCCC3)s2)=O)CCCCN(CCCC2CCOC2)C1 N1(C(C(OC)OC)=O)CC(C2CCCCN(C(c3ccc(Cl)c(F)c3)=O)C2)C1 CN1CCCC1(C)C(=O)NC1CC(N(C(=O)CCc2cccc(C(F)F)c2)C)C1 N1(C(CN(C(C)=O)C)=O)CCC(CCC(=O)N2CCC2C(C)(C)O)CC1 C=Cn1nncc1C(=O)NCc1cc(Br)n[nH]1.c12cn(nn1)C1CN(C1)C2=O c1(C(=O)NCC2(O)CC(NC(c3c(C)cccn3)=O)C2)ccc2nncn2c1 Cc1nc(C)c(CC(=O)NC2C=CCN(C(=O)CC3(O)CCOC3)C2)s1 CC1(C)CN(C(C2(O)CCCCCC2)=O)CC(C)(C)S1(=O)=O S(=O)(=O)(c1ccc(F)c(Cl)c1)N1CC(F)CC(C(=O)Nc2c(NC)cccc2)C1 C1(CC(C)NC(CC=C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 c1(C(=O)NCC2C(NC(c3cc(C)nc(C)c3)=O)C2)cccc2sccc12 c1(CN2CCC(=O)N(Cc3ccccc3)CC2)cc2cc3c(cc2[nH]1)OCCO3 C(=O)(CC1C(=O)Nc2c(F)cccc21)N(CCCN1CCCC1)C c1(C(=O)NC(CNC(c2c(C)coc2)=O)CO)ccc(-c2nnc(O)o2)cc1 C1(C(N(CCNC(C(CCC)O)=O)C(C)C)=O)CC2CCC(C1)N2 C12(CNC(CCCCCCC)=O)CCCCC1N(C(c1cc(C#N)c[nH]1)=O)CC2 Cc1csc2c(CC(N3CCCC3C(=O)N(C)C(C)C)=O)cccc12 N1(C(C(C)OCCCC)=O)CCC2CN(C(c3cc(C#N)ccc3F)=O)C(C)C12 c1(CC)ccc(OCC(=O)N(C)CC2(NC(C3CCC3(F)F)=O)CC2)cc1 C(=O)(CCCCCF)NC(C1CCN(C(c2ccc(CC)cc2)=O)C1)C Cc1ccnn1CC(N1CC(CNC(=O)C(F)C2CCC2)C1)=O C1(CNC(=O)Cc2ccon2)COCC1NC(C1(c2ccccc2)COC1)=O Cc1cc(C(=O)NC2CCN(C(=O)CCn3cccn3)C(C)C2)ncc1Br C1(F)(CNC(CCCOCCOC)=O)CCC(NC(C2CC(=O)N(O)C2)=O)C1 C1(C(=O)NC2CC(CNC(CNC(=O)NC)=O)C2)CCOC(C(C)C)C1 CC1CN(C(c2c[nH]nc2C2CC2)=O)CCN(C(=O)CSCc2ccncc2)C1 N1(C(c2c(OC)nccc2)=O)CCC(NC(c2csc(C)n2)=O)C(F)C1 N1(C(CCCCC)=O)CCCOC(CNC(c2n[nH]cc2Br)=O)C1 N1(C(CC2CCC(NC(c3cnc(C)s3)=O)C2)=O)CCC2(COC(=O)N2)C1 C(CN=C(NC)NC1CCOCC1)CC1(C)OCCO1.C1(C(=O)N)CCC=CO1 C(=O)(C1Cc2ccc(F)cc21)NC1CC2(CCCN(C(CC(CC)(C)C)=O)C2)C1 C1(NC(CC(C)C2CC2)=O)CN(C(c2sc(N(C)C)nc2Cl)=O)CC2CC12 c1(C(=O)NC(C2CCCN2C(c2cnc(S)[nH]2)=O)(C)C)nc2ncccn2n1 C#Cc1nccnc1NC(C1CCCCC1NC(c1ccon1)=O)=O c1(C(=O)NC(CC)CNC(c2n[nH]c(O)n2)=O)ccc(C)c(Cl)c1F C(N=c1nc(C2CCC2)[nH]s1)c1c(C)cc(F)s1 c1(NC2C3CN(C(CCOC)=O)CC32)ccc([N+](=O)[O-])c(C(F)(F)F)c1 CC1(C(=O)NC(CNC(C2CCCN2N=O)=O)C2CCC2)CS(=O)(=O)C1 C1(C(C(=O)NC(C2CSC2)C)C)CCCN(C(=O)OC(C)(C)C)C1 c1(NC(N2CC=CC(NC(C3C(CC)C3)=O)C2)=O)c[nH]c2ncc(Br)cc12 CC1CCC(NC(=O)C(C)(C)C(F)F)CN1C(=O)CCOc1ccc(Cl)c(Cl)c1 C1(NC(c2ccc(=N)[nH]c2)=O)CCN(C(c2scnc2C2CC2)=O)CC1C(N)=O C(=O)(C(CNC(C1CC1(F)Cl)=O)C(C)C)N1CCC(CCC)C1 CC1CC(C(=O)NCC2CCC3(CC2)CC3)CCN1C(C1CC2(CC2)CO1)=O C1(CC=C)(C(=O)NC2CCC2C(=O)OC)CN(C(=O)CCCNC(C)=O)C1 Cc1cccc(C)c1C(=O)NC1CC2(C1)CC2NC(=O)CC1CC2(CC2)C1 C(=O)(C1=CC(O)CCC1)NC1CN(C(C=Cc2ccc(OC)cc2)=O)CC12CC2 c1(OC)ccc(C(=O)NC(C)COCC(F)(F)F)c(Br)c1F c1(N2CCC(NC(CC)=O)(CF)C2)cc(C)nc(C(C2CC2)OC)n1 C1(NC(C2COCCOC2)=O)CC2(CCC2)C1OCc1ccccc1 C1(CN2CCC(NC(c3c(C(=O)OC)c(C)[nH]n3)=O)C2)CCC(F)(F)CC1 CC1(C)CCCC(C(=O)NCc2ccccc2CNC(=O)CCCCO)C1 N1(C(C2CCCN(C)C2)=O)CCC(C(=O)NCc2ncc(F)cn2)C1(C)C C1(NC(CC)(CC)c2nnnn2C2CCC(C(=O)OC)C2)CCCCC1CO C#Cc1ccnc(C(=O)NCCN(C(=O)CCc2nncs2)CC(C)O)c1 N1(C(c2c(C)nc(C(C)C)o2)=O)CCOCC(NC(=O)C(C)(O)C(C)C)C1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)CN2C(=O)CCC2=O)C1 c1(NC(c2nc(CNC(CC3C(C)OCC3)=O)cs2)=O)c(F)ccc(F)c1Cl C1(CNC(CC(CC)C2CC2)=O)CCC2(CN(C(c3cc(CC(C)C)c[nH]3)=O)C2)O1 CC1(C)CC=C(C(=O)NCC23CCC2CN(C(c2ocnc2C2CC2)=O)C3)CC1 C(CCCCNC(C12CCC1CC2)=O)NC(=O)CCn1ccnn1 CC(C)(O)CC(=O)N1CCCC1CNC(c1cccc(C2CNC(=O)C2)c1)=O C1(F)(CNC(=O)Cc2cnccn2)CCCN(C(=O)CSCC(F)F)CC1 N1(C(c2n(CC)nc(C)c2)=O)CC2CCN(C(c3cnn4ccccc34)=O)CC12 c1(OC)cc(C)cnc1C(N1CCCC(CNC(=O)C(O)CSC)CC1)=O C1(NC(CCC)=O)CC(CNC(=O)C(N2CCNC(=O)C2)C)C(O)C1 N1(C(c2c(C)cc(Cl)cc2)=O)CCC(C2CCOCC2)C1 C(=O)(C1=NN(c2ccccc2)C(C(N)=O)C1)N(C(c1ccco1)C)CC C(=O)(C(C)(F)C(C)(C)F)N1C(C)CN(C(c2c(F)cccc2Br)=O)CC1 C(=O)(C(C)CCCC(C)C)N(c1c(C)ccc(OC)c1)C.C1(=O)CC(C)(C)CN1 Cc1ccc(CNC(=O)COC2CN(C(c3ncccc3N)=O)C2)c(F)c1 C1(CCOC)CN(C(c2cnsn2)=O)CCN1C(=O)CC1(C)CCC1 CCCC(C)(CC)C(=O)N1CC(C)C(C)(C(=O)N(CC(=O)OC)C)C1 N1(C(c2cc(CC)on2)=O)CC(F)(F)CC1CNC(C1CC12CCC2)=O c1(C(=O)NCC=C)ccc(C(N2CC(NC(c3ccc(C)o3)=O)C(C)C2)=O)cc1 CN1CC=CCC1CC(=O)NCCCCCCNC(C1(C)CC2CC2C1)=O c1(NCC(N2CCC(CNC(COC)=O)CC2C)=O)ccc2ccccc2c1 C=CCC(CC=C)NC(C1CC(N(C(=O)CCC(C)SC)C)C1)=O CCCC(C)(O)CC(=O)NC1C=CCC(C(=O)NC2CCN(C(C)C)C2)C1 C(=O)(C1=COCCO1)NCCCN(C(=O)CCc1c(F)cccc1F)C C1(CCC(=O)NCCCN(CC(=O)NCCCC)C)CCCCCC1 C1(CC(N2C(C3(C)CCN(C(CCCC)=O)C3)CCC2)=O)CC2CCC(C1)N2C Cc1nnc(CC(=O)NC(C)(CNC(=O)C(F)(F)c2cnn(C)c2)CO)o1 c1(C(N2CCC(C(C)NC(c3ccccc3)=O)C2)=O)ccc(NC(C)=O)s1.C(C)(C)(C)N N1(C(=O)CC2CCC2)CCN(C(=O)CC2CCCC2)C(c2ccncc2)C1 C(CC(C)C(=O)NCC1(NC(c2cccnc2F)=O)CC1)OC c1(CN2CC3(CC(NC(C4CCC5(CCC5)C4)=O)C3)C2)cnc2n1CCOC2 Cc1cc(O)c(C(N2CC(N(C(=O)CN3C(=O)CCC3=O)C)C2)=O)nn1 C(=O)(N=c1ncn(CC(F)F)[nH]1)NCC(c1ccccc1F)(C)C c1(C(N(CCNC(=O)COCCOC)CC)=O)ccc(-n2ccnn2)cc1 C1(NC(CCC2N(C)CCC2)=O)CN(C(=O)CC2CCCOCC2)CC12CC2 N1(C(CCC=C)=O)CCC(C2CC2)C1CNC(c1ncn2cccnc12)=O C=CCC(C(=O)N(CCCNC(c1[nH]c(=N)sc1C(F)(F)F)=O)C)C(C)C c1(C(=O)NCC2N(C(C=C3CCN(C)CC3)=O)CC=C2)csc2nccn12 c1(CC)nc(C)c(C(N2CCC(C(C)NC(c3cnn(C)n3)=O)CC2)=O)o1 c1(C(=O)NCC(C)CN(C)C(c2ncc(F)cn2)=O)ccc(N)c(Br)n1 C1(CS(=O)(=O)NC2(C)CCOCC2)CN(Cc2ccccc2)CCCO1 C(N=c1nc2sccc2c(NCC2(C)COCCO2)[nH]1)C12CC(C)(C1)C2 C1(C(C)C)C(=O)N1.c1(OC)cc(C(=O)NC(CC2CCC2)CO)on1 c1(C(=O)NC2CC(CCNC(c3c(C)con3)=O)C2)cnn(CC(C)C)c1C C1(NC(C2N(C)C(=O)CCC2)=O)CCC2CCN(C(C3(n4ccnn4)CC3)=O)C12 C1(NC(C(=O)NC2(c3cccc(C)c3)CCCC2)=O)CCCNCCC1(F)F N1(Cc2cccc(N(C)CC)c2)CCC2(CCCOC2)C1 CC1(C)CC(CNC(C2C=CCCN2C(=O)CCc2csnn2)=O)CC1 c1(C(CCC(=O)N(CC(CCC)O)C)=O)cc2ccc(N(C)C)cc2[nH]1 c1(N(C)C)ccc(N)c(C(=O)NC2C3CC2CN(C(C2CC4CC2CO4)=O)C3)c1 N1(C(C2C3CN(C(CC4C(C)C(=O)CC4)=O)CC32)=O)CCCC2(C1)OCCCO2 C(=O)(C(F)CC(C)(C)C)NCc1cc(C(N2CCCC(C=C)C2)=O)sc1 Cc1cc2n(n1)CCN(C(=O)Cc1ccc(-c3ccccc3)cn1)C2 c1(C(=O)NCCN(CCOC)C(C2CCCCC2OC)=O)c(C)cnn1C N1(C(CC(C)C)=O)CCC(CNC(c2cnc(Cl)c(F)c2)=O)C12CCC2 c1(OC)nccc(C(=O)NC2CCC2NC(c2sccc2C(C)C)=O)c1F N#Cc1c(F)cc(C(=O)NCC2(NC(c3cnc(O)o3)=O)CC2)cc1F C1(C(=O)NCC(CCO)OC)CCCN(C(C23CSCC2C3)=O)CC1 c1(C(C(=O)NCC(CC)(C)NC(=O)C(=O)N(C)C)C)ccc(Cl)cn1 C(C1(C)CCOCC1)=CC(=O)NCC(C)CNc1ncc(Br)cn1 c1(N2CCCC(CC)C2)nc(C)ncc1F.c12ccccc1CC(=O)NC2C CN(C)S(=O)(=O)NCC(N1CC=CC(NC(C2CC2c2ccccc2)=O)C1)=O CCCCC(CNC(c1cc(C2(Cl)CC2)n(C)n1)=O)NC(c1c[nH]nc1CC)=O C(=O)(C1CCCc2ccccc21)N1CCC(C)(NC(C(C(C)C)O)=O)CC1 C1(CC)(NC(=O)C=CC(C)(C)C)CCN(C(=O)CCS(N)(=O)=O)CC1 c1(CC)nc(COC(F)(F)F)n(-c2cccnc2OC)n1 C1(NC(CN(C)CC)=O)CCN(C(=O)CN2CCOCC2=O)C(C2CC2)C1 c1(NC2CC(NC(c3c(SC)c(F)ccc3)=O)C23CCC3)ncc(C#N)cc1F N1(C(C2(COC)CC2(F)F)=O)CCC(F)(CNC(c2cccnc2C)=O)CC1 C1(C(=O)NCC2N(C(c3c(C)cncc3)=O)CC(O)C2)CCCCC1(F)F Cc1cc(C(N2CCCC(CN(C)C(C3CCCS3(=O)=O)=O)C2)=O)cc(C)c1 Cc1c(C(C2CC2)NC(=O)C(=O)N(C)C(C)C)cnn1-c1ccncc1 N1(C(c2cnn(C(C)C)c2N)=O)CCC(NC(=O)CC(C)n2cccn2)C(O)C1 Cc1cc(C(=O)NCC(Cc2ccccc2)NC(=O)C=CCO)cn1C(C)C C1(n2cnnn2)(C(=O)NC2C(NC(=O)CC(O)C3CCCC3)CC2)CCSCC1 Cc1cc(O)ccc1CC(N1CC2CC2(NC(=O)CCN(C(=O)CO)C2CC2)C1)=O C1(C(=O)NC2(CO)CC2)CC2(CC2)CN1C(=O)CC1CCCOC1 N1(C(Cc2ncc(C)[nH]2)=O)CC(CNC(c2ccc(Cl)cn2)=O)C(C)(C)C1 CCCCCCCCCCCC(=O)N1CC2CC1CN(C(=O)CC=C(Cl)Cl)C2 c1(C(=O)NC2(CO)CCN(C(=O)Cc3cccnc3)CC2)nccn2cnnc12 C1(CC(=O)OC)CCCN(C(N2CCC3(CC2)CC3)=O)CC1 c1(C(=O)NCCCC)ncccc1Sc1cccs1.C12CCN(C1)C(=O)CS2 c1(C(CC)NC(=O)NC(C)CN(C)C)ccc(-n2ccnc2)cc1 CCC1=C(C(=O)NCC2CCN2C(=O)CC(C)OC)CCCO1 C(=O)(CCCCC(C)(C)C)N1CC(C(C)NC(=O)CN2C(=O)CCC2=O)C1 N1(C(=O)CCn2cc(CCC3CCCOC3)nn2)CCC(c2ncon2)CC1 C1(CNC(CC)=O)CN(C(c2ccncc2-n2cccn2)=O)CC1(F)F C1(NC(C(C)(C)OC(C)=O)=O)CC2OC(C)(C)OC2C1.C12(C)CCCN1C2=O N#Cc1ccc(C(N2CCCC2C2(NC(c3cccc(C(F)F)n3)=O)CC2)=O)o1 N1(C(C2CN3CCC2C3)=O)CCC2(C1)CN(C(C1CC(O)CCN1)=O)C2 C1(C2CCN(C(=O)CNC=O)CC2)(C(=O)NCC(CCC)O)CCOCC1 C12(NC(=O)CCCc3nccs3)CCCC1(F)CN(C(=O)CCn1cncn1)C2 c1(C(=O)NC2CCCC(CNC(=O)C=C3CCCCC3)C2)c(F)ccc(F)c1O c1(C(N(C(CC)C(=O)NOC2CC2)C)=O)cc(C)c(C)cc1C C(=O)(C1Cc2ccccc21)N1C(C(=O)NCC(C(CC)C)CO)CCC12CC2 Cc1ccc(CN2CC(C(=O)NCCNC(c3ccnnc3O)=O)CC2=O)cc1 C1(CNC(C2CC(OC)C2)=O)CN(C(c2cc3ccsc3s2)=O)CC(C)(C)O1 c1(C(N(C(C(N2CC(C)CC(CC)C2)=O)(C)C2CC2)C)=O)c[nH]c2nccc-2c1 C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C(CNC(c2ccc(OC)c(C)c2)=O)CC1 N1(C(c2cnc[nH]2)=O)CCC2CN(C(c3c(OC(F)F)cccc3Cl)=O)C2C1 c1(OC)cc(F)c(C(N2CCC2(C)C(=O)Nc2sc(C)cc2C#N)=O)cc1OC C1(C(=O)NC(C)Cc2cccc(Cl)c2)CCC(=O)CC1C C1(C)(CC)CC(NC(=O)CSCC(N)=O)CN1C(c1cccc(Cl)c1)=O c1(C(N2CC(CSC)OCC2)C(=O)NCC2CC2)ccc2ccc(F)c(F)c2n1 N12CCCC(C1)C2.O=C1CCC(C(N2CCN(C(C3CCCO3)=O)CC2)=O)CN1 Cc1cnn2ccc(C(N3CCCC4(NC(=O)CCC(F)F)CCCC34)=O)nc12 c1(C(N2CCCC3CN(C(C4(C5CC5)CC4)=O)CC23)=O)[nH]nc2ncnc(O)c12 c1(N(CC#CC)C)nc(=NCC2CCC(F)C2)nc(N2CCOCC2)[nH]1 CC1COCC1(CO)NC(c1nnnn1C1(C)CC1)c1csnn1 C(=O)(C(C)C(CC)CC)N1C(CNC(C2(C=C)CCOCC2)=O)CN(C)CC1 C(C(N=[N+]=[N-])C(=O)N(C)CC1CN(C(c2cc(C)cnc2C)=O)C1)OCC C(CCNC(c1ccc(O)nn1)=O)(C(=O)N1CC2CC2C1)OC c1(-c2nn(-c3ccn(CC)n3)c(C3CC3(C)C)n2)cc(F)c(N)c(F)c1 CC1CCC(C(F)(F)F)CN1C(c1ccc(CC#N)cc1F)=O C1(C(=O)NC2CCC(NC(C3CC3c3cccs3)=O)C2)(CO)CC(F)(F)C1 C1(n2cc(C(C)(C)O)nn2)CN(C(C2CCCC(=O)CC2)=O)CCC12CCC2 C(CCOCCO)(C(=O)NC(c1ccn(C)n1)C)NC(C(CN(C)C)O)=O c1(C(N2CC(CNC(CCC=C=C)=O)C3(C2)CCC3)=O)nc2nc(C)ccn2n1 c1(CC)ccc(C(N2CCC(C)C2CNC(c2cccc(C3CC3)n2)=O)=O)cn1 Cc1cccnc1C=CC(=O)NC1(CNC(c2ccnn2C)=O)CCCCC1C N1(C(CSC2(C(N3CC(C(N)=O)C3)=O)CC(=C)C2)=O)CC(F)(F)CC1C C#Cc1cc(C(=O)NCC(C)NC(=O)C(C)(O)COC)ccc1C C1(C(=O)NC2(CCNC(c3cncn(C)c3=O)=O)CC2)CCC2(C1)CC2(F)F N1(CC(N2CCC(NC(CC3(OC)CCC3)=O)CC2C)=O)C(=O)NC(C)(C)C1=O C12(NC(CN(CC)CC)=O)CCCN(C(=O)CCCCN3CCOCC3)CC1C2 c1(NC(C(OC)OC)C)ccc(S(=O)(=O)NCCCc2nccs2)c(Cl)c1 Cn1ccc2cc(-c3n[nH]c4c3CN(c3ncc5cn[nH]c5n3)C4)cnc12 c1(C(=O)NC2C(O)CCN(C(CCOCC#C)=O)C2)ccc(OC)c(OC)c1C C(CCCC(C)NC(=O)Cn1ccsc1=N)NC(C=C(C)Cl)=O c1(C(N(CC(C)NC(=O)CCOCC)CC2CC2)=O)csc(Cl)c1Cl C1(C(=O)NCCCN(C)C(c2nnc(O)cc2O)=O)CC2(CCCC2)C1 c1(OCC=C)ccc(Cl)c(C(N2CCCC(O)(CNC(c3ccc[nH]3)=O)C2)=O)n1 C1(CC(C)NC(N)=O)CCN(C(C2CN(C(C3(c4cccs4)CC3)=O)C2)=O)CC1 N=c1ccc(C(=O)NC2C=CC(CNC(c3cn(CC(F)F)cn3)=O)C2)n[nH]1 c1(NC(C2CS(=O)(=O)CC2N2CCOCC2)=O)nc2cccc([N+](=O)[O-])c2s1 c1(C(C)NC(C(=O)NCCCC)CC)ccc(OC)cc1 c1(C(=O)NC(CNC(C(C=C)(C)C)=O)(C)CO)cc(C)cc2c1NCCC2 Cc1cccc(N)c1C(=O)NC1CC(O)CN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCC2C(C(F)(F)F)CCN(C(CSC)=O)C2)CCc2nn[nH]c2C1 Cc1cc(C)c(CNC(=O)COCCN(C(=O)CCC2CCC2C)C2CC2)s1 c1(OCC(=O)NCC(C2CC2)NC(Cc2c(C)ccnc2)=O)ccc(Cl)c(F)c1 N1(C(c2cc(C)no2)=O)CC2CC(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 c1(C(N(C2CCN(C(c3c(Cl)cccc3Cl)=O)CC2)CC)=O)ccc2c[nH]nc2c1 CC(C(=O)NCCSC(C)(C)C)C(C)NC(c1nccnc1O)=O c1(CC(=O)NCC2CN(C(C=CCOC)=O)C3C2C3)c(C)nn(C)c1Cl C1(C(=O)NCC2CCN(C(CCC(=C)Br)=O)CC2)CCC(C)(O)CC1 c1(CNC(C2CC(C(=O)NC3(C(F)(F)F)CCC3)C2)=O)cc(I)ccc1F c1(CCC(=O)NCCCN(CCCNC(C2CC23CC3)=O)C)ccnn1C C(=O)(C(C)CC(C)(C)C)N1CCC(=C)CC1C(=O)NCCc1nc(C)oc1C Cn1c(=O)oc2c(C(N3CCCN(C(=O)CNC=O)CC(O)C3)=O)cccc12 CCCCCC(C(=O)NCC1CCN(C(=O)C(C)C2CCC2)C1(C)C)C(C)C c1(CC(=O)N(CCN(C(C2CC2C)=O)CC)CC)ccon1 Cn1cc(S(N)(=O)=O)cc1CC(=O)OCc1ccc(OC(F)F)cc1 N1(C(COc2cc(C)on2)=O)CCC(C)CC1CNC(=O)C(C)NC(N)=O C1(NC(C2C(CCC)C2)=O)(CNC(=O)C(O)CN2CCOCC2)CCCCC1 C1(NC(CCCC#CC)=O)CCOC12CCN(C(=O)CC1NC(=O)NC1=O)CC2 Cc1ccc(C(=O)NCC2CC(NC(=O)CC3CC(F)(F)C3)C2)cc1Cl C1(N(C(c2c(C)snc2)=O)C)CC2CC1N(C(c1cccn1C)=O)C2 N1(C(c2ccc(C#N)cc2)=O)CCN(C(C2CCSCC2)=O)CC(O)C1 CCC(C)C(C)C(=O)N(C)CC1(O)CN(C(c2ccc(SC(F)F)cc2)=O)C1 Cn1cccc(C(=O)NC2COCC2NC(=O)CC2(C)CC2)c1=O N1(C(C(=O)NCCC(=O)OCC)C2CC2C)CCCOCC1C N1(C(C(CC2CCOCC2)NC(c2c(C)scc2)=O)=O)CC(CO)C1(C)C CSC1=C(C(=O)NCCC2(O)CCCN(C(C3CC(O)C3)=O)C2)CCCC1 c1(Nc2ncc(C(N3C(C(=O)OCC)CC(C)CC3)=O)s2)n[nH]c2c1CC1CC21 c1(-c2nc(C)nn2-c2cn[nH]n2)c2c(nn1C)CCC2.c1(C)n[nH]c2cccnc12 c1(CC(=O)NCC2CN(C(c3cc(O)no3)=O)CCCO2)n[nH]c2c1CCCC2 C1(CC)C(NC(=O)CS(=O)(=O)NC)CCCN1C(=O)C(C)c1cc[nH]n1 c1(SC(C(=O)NCC(CNC(CC(CC)OC)=O)C)C)ccc(Br)c(C)c1 N1(C(C(c2cccnc2)C)=O)CCCCC(NC(c2ccccc2C2CC2)=O)C1 CN1CC(C(N2CCOC(CC(=O)NC34CC3COC4(C)C)C2)=O)CCC1=O CC1CC(NC(=O)Cc2ccc(F)c(F)c2)CN(C(c2cc[n+]([O-])cc2)=O)C1 CCC(CCCC(=O)NC1CCCC1(C)O)NC(c1ncccc1F)=O N1(C(CCN(C(=O)CCc2cncs2)C2CC2)=O)CC2(CCCO2)C1 C1(NC(c2ccc(Cl)cn2)=O)CCN(C(c2csc(Cl)n2)=O)C12CC2 CC1OCCC1(F)F.C12CCN(C(=O)OC(C)(C)C)C1CN2 c1(CC(N2CC3CC2CN3C(c2cnc(O)cc2O)=O)=O)c(Cl)cc(Cl)cc1Cl c1(C(=O)NC(CNC(C=C(C)Cl)=O)CO)cc2cc(C)ccc2[nH]1 C(=O)(CC(C)C(=O)NC(c1ccccc1)C(N1CCC(F)(F)C1)=O)OC C1(O)(CCNC(C(C)N2CCC2)=O)CCCN(C(c2cc(=O)c(O)c[nH]2)=O)C1 C(=O)(CC(C(F)(F)F)C1CC1)N(CC(C)(C)CNC(=O)Cc1ccsc1Cl)C N1(C(CCOCC)=O)CC(NC(=O)C2=C(Cl)CC2)C2CC12 CC1(F)CN(C(=O)CN2CCOCC2)CCN(C(C2(C(F)(F)F)CCCC2)=O)C1 C1(C2(NC(C3CCN(C(=O)c4ccon4)O3)=O)CC2)(OC)CCC1 N1(C(c2c(C)occ2)=O)CCC(C)(C)C(C(=O)NC(C)(C)CCF)C1 N1(C(CC(CC)NC(CCCC#C)=O)=O)C2CCC1COC2 CC1=CCCN(C(C2(F)CN(C(=O)CC3CCCC(C)O3)C2)=O)C1 c1(OC)ccccc1CC(C)(C)C(=O)NCC(CNC(=O)CSC1CC1)CO c1(CNC2(c3n(C(C(=O)OC)C)nnn3)CC(C)C2)c(Cl)c(C)nn1C Cn1ccc2cc(C(N3C4CCC3CN(C(C3CS(=O)(=O)C3)=O)CC4)=O)ccc12 C(=O)(CCS(=O)(=O)CC(C)C)Nc1ncnc(C)c1C.C12CN(C)C(C)(C1)C(=O)O2 C(=O)(C(C(C)(C)C)C1CCC1)NC1C(C(=O)NCc2ccc(OC(C)=O)cc2)C1 N1(C(c2c(OC)scc2)=O)CCN(C(=O)C(C)OCC(F)(F)F)CCC1C C1(c2c(C)ncc([N+](=O)[O-])c2)NC(=S)N(C2CC2)C2=C1C(=O)N(C)C2(C)C C(CN(C)C)(C(=O)N1CC(CC2CC2)C1)NC(CC1C(C)C1)=O C1(C(N(CC(OC)OC)C)=O)C=CCCN1C(C1CCC(C)(C)C1)=O C1(C)(C(=O)NCC(C)N(C(=O)C=CCF)C)C=CCCC1 CC1CC(C)C1C(=O)NC1(CN(C)C(c2ccc(OCC(F)(F)F)o2)=O)CC1 N1(C(C2CC(CCC)OCC2)=O)CC=C(CCNC(c2cn(C)cc2C)=O)CC1 C1(NC(CSCCOC)=O)CN(C(=O)CCCC2CCCCC2)C(C)(C)C1 C1(CN(C(C2(COC)CCC2)=O)C)CCN(Cc2ccccc2)C1 C1(CNC(=O)CCN2CCCC2)C(C2CC2)CCN1C(c1nc(O)[nH]c(=O)n1)=O C=C1Cn2c(C(N3CC4CCC4(NC(C4CC4(C)CC)=O)C3)=O)nnc2S1 c1(CCC(=O)NC2CC(NC(COC(CC)C)=O)C2)ccc(F)cc1Br C1(NC(c2cc(C)n(C(C)(C)C)n2)=O)CC(C)CN(C(c2ccc(O)cn2)=O)C1 Cc1cc(C(N2CCCC(C(=O)NCC3CC(F)(F)C3)C2)=O)cc(C)c1F c1(OC(C)C)ccccc1CC(N1CCC(C(CO)NC(=O)CCCF)CC1)=O c1(C(N(CC(CC)O)C)=O)cccnc1CNC(=O)COCCCF c1(C2(C(N3CC(NC(C)=O)(CO)C3)=O)CCCC2)cccc(C)c1 CC(C)C(C#N)C(=O)NC(C)(C)CNC(c1ccc(C(F)(F)C(F)F)cn1)=O N1(C(c2c(OC(F)F)cc(C)s2)=O)CCN(C(C2CC(C)C2)=O)CC(O)C1 c1(C(=O)NC2C(C)(C)N(Cc3ccccn3)CC2)noc2c1COCC2 CC(C)CCCC(=O)NCC1CN(C(=O)C2=CCCOC2)CC1O C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C(C(C)C)NC=O)=O)CC1C C(CN=C(NCC1CCCO1)N1CCOC(C)(C#N)C1)c1ncc(C)cn1 Cc1nocc1CNC(=O)C(C1CCC1)NC(=O)C(C1CC1)SC Cc1c(C(N2CCC2CNC(=O)CC(C)C(C)(C)C)=O)cc(S(N)(=O)=O)cc1F C=C(CNC(=O)CC(C)C(C)(C)NC(=O)Cc1cnc(C)s1)c1ccccc1 N1(C(C2CCC2)=O)CCC(C(=O)NC2CCC(NC34CCC3C4)C2)CC1 C12(C(N(C3CCN(CCc4nc(C)on4)C3)C)=O)CCC(CC1F)C2 C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(C(=O)CSc1ccc(OC)cc1)C2 C(=O)(CCS(N)(=O)=O)N1CCC(C(C(=O)NCC(CC)(C)CC)F)C1 C1(N(C(=O)NC(c2noc(C)n2)CC)C)CCCN(c2cccc(F)c2)C1 c1(C(N2C(CN(C(C(n3cc(Cl)cn3)C)=O)C)CCC2)=O)nnn(C)c1N C1(NC(C(C)SC(C)C)=O)(CNC(=O)CCC2CCCCO2)CCOCC1 N1(C(C2(NC(c3cnn[nH]3)=O)CC(CO)C2)=O)CCCNC(=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)NCC(CCNC(C1CCCCNC1=O)=O)O CCC(C)(COC)C(=O)NCC(C)(C1CCC1)NC(=O)COCCOC C(=O)(C(C)C(C)C)NCC1C(NC(c2nc(CCC)oc2)=O)COC1 c1(NC(C2CN(C(=O)CCc3cccnc3)C2)=O)cnc(O)c2ccccc12 CC1CN(C(C2CN(C(c3cc(CCO)on3)=O)CC2(C)C)=O)CC1(C)CO N1(c2c(Nc3c(OC)ccc(OC)c3)nccc2)CCC2(C1)OC(=O)NC2C C1(C(N(CC=C)CC)=O)CC(O)CN1C(C1CCNC1=O)=O Cc1cnc2n1CCC(C(=O)NC1(c3cccnc3)CCOCC1)C2 Cc1ccc(O)c(C(=O)NCCCCCCNC(c2cc(C)[nH]n2)=O)c1 c1(COC)nn(C)cc1C(=O)NCC1C=CCN1C(=O)C(O)COC N1(C(c2n(C)nc3c2CCC3)=O)CC2(CCN(C(C3C4CC(=O)CC34)=O)CC2)C1 c1(CNC(C(CNC(=O)CC23CCCC2C3)O)=O)n[nH]c2c1CCC2 Cc1cc(C(=O)NC2CCOC(CNC(=O)CCCC3CCOCC3)C2)[nH]c1C CCC(C)(C)C(=O)C(=O)N1C(C(=O)O)CCC1C1CCC1 C(C(O)C(=O)NCCCN(C(=O)CC1CC1)CCO)=CCCC N1(C(C2CN(C)C2)=O)CCN(c2ccc(C(F)(F)F)nn2)C(CC#N)C1 c1(C(=O)NCCN(C(C(C)OCC#C)=O)CCOCCO)c(Cl)n[nH]c1CC C(Cn1ccnn1)(C(=O)NOCCF)NC(C1CCNC1=O)=O c1(C(=O)NC(C)C)ccc(C(=O)NC(C)(CNC(C2C=CCC2)=O)C(C)C)cc1 c1(COC(CC(c2ccc(C)cc2)C)=O)cccc(O)c1C C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(=O)CNC(c3cscn3)=O)CC2)C1 CN1CCN(C(=O)C(F)C2CCOC2)C(CNC(c2cc(O)ccc2F)=O)C1 C1(C(=O)NC23CC(C(=O)NCCN(C)C4CC4)(C2)C3)CCC(C2CC2)C1 c1(C2C(C(=O)NC(C3CCCC3)CNC(=O)C=CC3CC3)C2)cccnc1 N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(NC(=O)C(C)COC(C)=O)C1 C1(CNC(c2cccc(C(C)C)n2)=O)CN(C(=O)C(O)CC(N)=O)C2(CCC2)C1 c12cccc(c1)CS(=O)C2.Cc1nccn1CCN(C(=O)C(=O)NC(C)C)C N1(C(c2n(CC)ncc2)=O)CC(NC(=O)Cc2nonc2C)C(C(F)F)C1 C1(NC(C(C)C2CCC2)=O)CN(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CC1(C)C c1(Cc2cc(CNC(C3CC(SC)C3)=O)n[nH]2)ccc(Cl)c(C(F)(F)F)n1 C(=O)(C(C)(C)c1cccnc1)NCCCN(CCCNC(=O)C(O)C1CCC1)C c1(C(N2C(C)(C)C(CNC(=O)Cn3ccnn3)CC2)=O)ccc(N)c(F)c1F Cc1[nH]c2ncccc2c1C(=O)NCC1CN(C(=O)C(C)CS(C)=O)CCCO1 c1(N2CCC(N3CC(C)(C)C3)CC2)nc2c(c(=NCC(Cl)Cl)[nH]1)CCCCCC2 N1(C(C2N(C(C)C)C(=O)CC2)=O)CCCC(O)(CCNC(c2ccnnc2)=O)C1 C#CCCCC(C)C(=O)NC(C)(CNC(c1noc2ncccc12)=O)CC C12(CNC(CN(C3CCC3)C)=O)CC(CO1)N(C(=O)CCc1n[nH]c(=N)s1)C2 c1(CNC(C2CC(CCC)C2)=O)nc(C(=O)N(C2CCCC2C)C)c(C)o1 CCC(CC)C(=O)NCc1ccccc1.C(C)(C)(CC(N)=O)N(CC1C(=O)N1)C N1(C(CC)=O)CCc2cc(-n3c(=O)c(=O)nc4nc3NS4)ccc21.C(C)(=O)OC N1(C(CC2CCC(=O)O2)=O)CCCC(NC(=O)COCc2cccnc2)C1 c1(C(N2CCC(C(=O)NCCCC(=O)OC)CC2)=O)cc2ccccn2n1 C1(NC(C2CCC2(OC)OC)=O)CCOCC1.c1(C(=O)OCC)nonc1C1CC1 c1(OC)cncc(C(=O)NCC2CC(NC(c3cc(CN(C)C)cs3)=O)C2)n1 C1(C(=O)NC2(COC)CCCCC2)COCCN(C(C2(C)CC2(C)C)=O)C1 N1(C(CC2CC(OC)C2(C)C)=O)CCC(NC(c2cc(Cl)n(C)n2)=O)C(C)C1 N1(C(c2[nH]cc(C)c2)=O)CCC(C)(C)C1CC(=O)NC(c1nnc(O)o1)C N1(C(C(N2C(c3ccc(C(=O)OC)o3)CC3CC32)=O)=O)CC2(CCOC2)C1 CC1(NC(=O)CC2CC=CCC2)CCCN(C(c2nn[nH]c2Cl)=O)C1 c1(C(=O)NC(C(C)NC(CCNC(C)=O)=O)C)cccc(OCC(=O)NC2CC2)c1 C1(C(=O)NC(C)C(C)(C)CO)(NC(c2oc(C)c(CO)c2)=O)CCC(C)(C)C1 n1(CC(=O)OCC)cc(C(=O)NCC(O)CN(C(=O)C(C)n2ccnc2)C)nn1 N1(NC(N(C)C(C2CC2(F)F)C2CC2)=O)CCCC(N(S(C)(=O)=O)C)C1 N1(C(C2(C)CCCC2)=O)CCCC(C2CCN(C(=O)COC(F)F)CC2)C1 C(=O)(C1=NOC2(CCNCC2)C1)N(CCN(CCC1CCC(C)O1)C)C C(CCCC(=O)N(CC(C)O)C1CC1)N(C(c1n(C(C)C)cnc1)=O)C Cc1c(C(=O)N(CCC#N)CCO)cccc1-c1nn[nH]n1 C(CC(F)F)(C(=O)Nc1cc(C(N)=O)cc(C)c1)N(C(c1n(C=C)nnc1)=O)C c1(NC(=O)COc2ccccc2)nnc2ccc(Cl)nn12.CC12CN(C1)C2=O C#CCC(O)C(=O)N(C1CCCN(C(=O)Cc2coc(-c3ccccc3)n2)C1)C CC1(C(N2CCC(CNC(c3cc(F)ccc3Cl)=O)C2)=O)CCC(F)(F)C1 CC1CCC(NC(=O)C2=CCCOC2)CN1C(=O)CN1CC2C=CC1C2 C1(CCC)CN(C(c2nocc2C)=O)CC1NC(=O)CC1CC=CCN1C C12(NC(c3ccc(CC)o3)=O)COC(C1)C(NC(=O)C(c1cscn1)N(C)C)C2 C(=O)(C(C(C)(C)C)N(C)C)NCC(C)(C)CC1CN(C(=O)CC(F)(F)Br)C1 N1(C(=O)CN2CCC2)CC2(CCN(Cc3c[nH]ccc3=O)CC2)C1 CC(C)(CC(=O)NCC1CCCN1C(=O)C#CC1CC1)C(F)F Cc1ccc2scc(C(N3CCCN(C(=O)CC4CC5(CC5)C4)C(C)C3)=O)c2c1 C1(C(=O)NCC(c2cn(CC)nc2)O)Cc2cc(C)cc(Br)c2O1 c1(C(N2C(C3(NC(C4CCOCC4)=O)CC3)CCC2)=O)cc2ccccc2[nH]1 c1(CNC(C(=O)OCC)Cc2ccncc2)cc(C)c(Cl)c(C)c1 N1(C(c2cncc(OC)n2)=O)CCN(C(=O)C=CC(C)(C)C)CC1CO O=S(=O)(c1cccnc1NCc1ccc(C2CC2)cc1Cl)N1CC2CCC1C2 c1(C(=O)NC(C(=O)OC)(C)C(F)F)ccnc2[nH]c(C(F)F)nc12 C(=O)(C=CS(C)=O)NCCNC(C1CN(C(C2C(C)OCC2)=O)C1)=O c1(C(N2CC3CC(NC(c4ccc(SC)s4)=O)C3C2)=O)c(C)ccc(F)c1N Cc1cccc(C(=O)NC2CCC(C(=O)N(C3CCCC3O)C)C2)c1O N1(C(c2n(C)nc(O)c2)=O)CCC(NC(=O)CO)C(CO)CC1 C(=O)(C1CCCc2occc21)NC(CNC(CS(CC(C)C)(=O)=O)=O)CO c1(CC)ccc(CCCC(=O)NCC(O)CNC(c2coc(OC)n2)=O)cc1 c1(C(=O)NCCC(=C)CNC(c2ccnc(O)c2)=O)cc(S(C)(=O)=O)ccc1O C(=O)(CC(C)(O)NC(N)=O)N(CCOCCN(C(C(C)CF)=O)C)C C1(NC(C=CCOC)=O)CCN(C(C2(C(=O)C3CC3)CC2)=O)CC1F CC1OCCC1C(=O)NCC1CCCC1NC(=O)CCc1nccs1 C1(C(=O)NC2(CCO)CN(C(CC(C)OC)=O)C2)COCCN1C1CCCC1 C(C(C(=O)N(C1CCNC1=O)C)C(C)C)NC(CNC(CCC)=O)=O c1(CC(=O)NC2CC(CCNC(c3cc(OC)no3)=O)C2)cc(F)ccc1F C(C)(CC1CCCCC1)(C(=O)NC(C)CCN(C(=O)Cn1nncc1C)C)OC c1(C(=O)NCC2(OC)CN(C(C3(C)CCCN3C)=O)C2)ccc(F)c(C(F)F)n1 c1(C(=O)NC(C2(CNC(c3cn(CC)nc3)=O)CC2)C)ccc2c(c1)CN(C)C2 CC(C)C(O)CC(=O)NC1CCC(NC(C2OCCC2C)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC(C)C3)=O)C2)n[nH]c2cccnc12 c1(OC)cccc(C(C)C(=O)NC2CCCCC2NC(c2cnc[nH]c2=N)=O)c1 CCC(C(=O)NCCCCNC(c1coc(C(C)(C)C)n1)=O)OC n1(CC(=O)NC2CN(C(C3(C(N)=O)CCC3)=O)CCC2F)cnc2c1CCCC2 c1(C(N2CC(NC(C(C)SCCCC)=O)(CO)C2)=O)c(C)cccc1F C=Cc1ccc(C(N2CC(N(C)C(C3CC(OC(F)F)C3)=O)C2)=O)cc1 CN1CCC(C)(C(=O)NC2(C)CCCN(C(c3nnc(O)cc3O)=O)C2)C1=O N1(C(C(C)CC2CC2)=O)CC(C(=O)NC(C)(C)CC2CC2)C(F)C1 CC(CC(=O)NC(C)(C)CNC(c1cnn(-c2ccccc2F)n1)=O)C(F)F C1(NC(c2c(COC)cc[nH]2)=O)(CO)CCN(C(=O)Cn2nc(C)cc2C)C1 C(=O)(CCC(C)C)NC1CCCC1.C1(C)CC(C)NC(=O)CN(CC)CC(=O)N1 C(=O)(CCCN=[N+]=[N-])NCC(CNC(C(CC)Oc1ccccc1Cl)=O)O N1(C(CCC#C)=O)CCC2(CC2C(=O)NOCC2CCCC2)C1 N1(C(c2nc(C)[nH]n2)=O)CCOCC12COCCN(C(=O)C=CCO)C2 Cc1ccc(C(N2CCC(C)C2CNC(=O)Cc2cc(Cl)ccc2F)=O)cc1Cl C(=O)(C(C)N=c1cc[nH]cc1)NCC1C(C)CCN1C(=O)C=Cc1cscn1 C1(COC)(NC(=O)Cc2ccsc2)CCN(C(c2cn(C3CC3)cn2)=O)C1 C#Cc1cccc(C(=O)NCC(C2(O)CN(C(=O)C=CC3CC3)C2)(C)C)c1C c1(C2c3cc2no3)[nH]c(=N)ccc1C.CC1=NOC(CNC(=O)NC)C1 CC1(CNC(c2cc(-c3ccccn3)ns2)=O)CCC(NC(C2CCC2)=O)C1 c1(C(N2CCC(N(C(=O)CCC(=O)C3CCCCC3)C)C2)=O)nc(Cl)ncc1Br CC1(C)CCN(C(C2CC23CCCCC3)=O)C1C(=O)NCC1=NOC2CCCC12 CC(C)(C(=O)NCC(O)C(=O)N1CCCC1CN=[N+]=[N-])C1CC1 c1(CNC(CC2(C)CCN2C(=O)COc2ccsc2)=O)n[nH]c2c1CCC2 C1(C(=O)NCC(C)C(=O)N(C)CCc2ccncc2)CCCCNC1=O N1(C(c2c(C)nc(O)nc2S)=O)CCN(C(c2cc(C#N)on2)=O)CC12CCC2 Cc1nc(C(=O)NCC(C2CCCC2)NC(=O)CN(C)C(N)=O)c(C(F)(F)F)[nH]1 CC(C(C)(C)N)NC(c1cnn(CC2CCC2)c1)=O.CCCCNC(=O)CC1CC1 C1(C2CCCC2)(C(=O)OCC)CCN(C2CC2C2CCC2)C1 N1(C(c2ccno2)=O)CC2COCC(C1)N2C(c1cc2cnccc2[nH]1)=O C(=O)(CC(C)(C)C=C)N(C1CCN(C(c2ccc(F)c(SC)c2)=O)CC1)CC#C C1(C(=O)NCCCNC(=O)OC)CCC2CCC1N2C(c1c[nH]c(C)c1)=O C#Cc1ccc(C(N2CCC(NC(c3cc(F)ccc3F)=O)C(O)C2)=O)cc1C Nc1cc(C(=O)NC2CC(O)CN(C(=O)C(F)=CCCF)C2)c(Cl)cc1Cl C1(C(=O)NCC#C)CCC2CCC1N2C(c1ncn(C)c1C)=O O=C1NC(c2cncc(CO)c2)C2=NNC(=O)C12 N1(C(CCOC(C)C)=O)CCC(CCF)(NC(=O)C(C)OC(C)(C)C)C1 C12COCC1C(=O)N2.N1(C(C(C)NC(=O)OC)=O)CCCC1c1ccco1 Cc1cc(-c2cn(C3CCN(C(c4c(C)ccn4C)=O)CC3)nn2)ccc1F c1(C(=O)NC(CC)CNC(=O)CC(C)(C)OC)cc(F)cc2cccnc12 C1(CC)CN(C(c2nnn(CC)c2C)=O)CCC1NC(=O)C(C)NS(C)(=O)=O Cc1cccnc1-n1ccnc1C1OCCC1Nc1nccnc1N C(=O)(C(C)(C)CC(C)(C)C)NCC12OCC(NC(C3N(CC)CCOC3)=O)C(C1)C2 C1(C(=O)NCC(C(C(=O)OC)F)C)CCN(C(C)=O)C(C)(C)C1 C=CCC(C(=O)NCC1CCC(C(=O)NC(c2cn[nH]c2)C)C1)C(C)C n1(CC)cnc2[nH]c(=NCc3cnc(O)nc3)[nH]c(=NC3CCOC3C(C)C)c12 c1(C(C)NC(C2(C)CCN2CC2CC(F)C2)=O)cccc(C(F)(F)F)c1F CC(C(=O)OC(C)(C)C)C(=O)N1CC2C(N(C(=O)CCCOC(C)(C)C)C)C2C1 C=CC1OCCC1C(=O)NCC1CC1CNC(c1ccc(SC)o1)=O N1(C(=O)NCc2ccc(Cl)cc2C(F)F)CCCC1C1CCCO1 c1(CC)cc(NCC2CCN(CCC3CCOCC3)CC2)ncn1 c1(CC(=O)NC(CCCNC(CC=C)=O)C)coc2cc(Cl)ccc12 c1(C(=O)NCCN(CCOC)C(c2c[nH]nc2Cl)=O)ccnn1C(C)(C)C c1(C(=O)OCCc2ccccn2)ccc(NC(c2ccon2)=O)cc1 c1(NC2CCN(C(Cn3ncc(C)c3)=O)C2)cc(O)nc(C)n1 c1(C(=O)NCCCN(C(C2C(C=C)OCC2)=O)C(C)C)cnc(O)c2cncn12 Cc1cccc(CC(=O)NC2CC2NC(=O)COc2cnc(Cl)cn2)c1 c1(C(N2C(Cc3cn(CCC=C=C)nn3)CCC2)=O)nn(C)c2ncccc12 C(=O)(C(CC)CCCC)NC1CC(C)=CCN(C(c2c(CC)ccc(C)n2)=O)C1 N1(C(C2OCCN(C(C)C)C2)=O)CC(NC(c2cc3sccc3[nH]2)=O)CC(C)C1 N1(C(CNS(C)(=O)=O)=O)CC2CCC1CN2C(=O)C(=O)NC(=N)N c1(C(=O)NCCC(C)N(C(=O)CCc2cncs2)C)cc(N)c(F)cc1F CC1CN(C(C2CCC3(C2)CC3(F)F)=O)CC2(CCN(C(C3CC3F)=O)C2)O1 N1(C(c2cc(OC)n[nH]2)=O)C(C)C2CC1C2NC(=O)CC1CCCC1 CN1Cc2ccccc2CC1C(N1CC(NC(C23CC(C2)C3)=O)C(F)C1)=O C1(=CC(N2CCC(N(C(=O)CCN3C(=O)CCC3=O)C)C2)=O)CN2CCC1CC2 C(=O)(C#CC(C)(C)CNC(=O)C(C)CC(C)C)NCCC(=O)NCC c1(CC)cc(C(=O)OCC2CC2c2ccc(Br)cn2)c(Br)s1 N1(C(C(C)(C)F)=O)CC2CCC1C(NC(C1(Cc3cnn[nH]3)CCC1)=O)C2 C1(CC)CN(C(=O)CC2C=CCCC2)CCC1NC(=O)CC1CC=CCC1 Cc1ncn2ccc(C(N3CCC(O)(C(C)NC(=O)CCCC4CC4)C3)=O)cc12 N1(C(CC(=O)OCC)=O)CCCCC1CN(C(=O)C(C)(C)COC)C c1(C(=O)NC2(CC=C)CN(C(=O)C(C)C3CC3)C2)ccn2c(C)cnc2c1 C1(C(=O)OCC)OCCNCC1N(CC(C)C)C(c1cnc(O)nc1O)=O C1(OC(C)C)CCCN(C(=O)CCCCN(C)C(c2c[nH]nc2C(C)C)=O)C1 N1(C(c2nc(C#C)sc2)=O)CCN(C)C(CNC(=O)CC(C)OC)C1 C1(C(N(CC(O)CN(C)C(c2n[nH]cc2[N+](=O)[O-])=O)C)=O)CCCCC(F)(F)C1 C1(C(=O)NCC2(F)COC2)COCCN(C(c2ccnnc2O)=O)C1 N1(C(C(C(C)C)O)=O)CCC(C2CC2)C1CNC(c1cccc2nsnc12)=O CCCC(CNC(c1cccc(O)c1F)=O)C(=O)N1CC(C)CC1CC C(C(C(=O)NCc1cnc(F)cc1C)C(C)(C)C)NC(C(CCCC)O)=O C(CCCCC(=O)NCC(C)C1CCC1)NC(Cc1c(C)noc1C)=O C#CCCCC(C)C(=O)N1CC2CCC1CC2NC(=O)CN1CCOCC1 C(c1ccccn1)=CC(=O)NCC1CC(F)(CNC(C2(C3CC3)CCCO2)=O)C1 C12(C(=O)NCC(C)CN(C(=O)C#CC3CCOC3)C)CCCN(CCC1)C2 C(=O)(C1=NOC(C)C1C)N1C(C(N(CC#C)CC2CCCO2)=O)C=CC1 C(=O)(C(=O)C(C)(C)C)N(CCC(=O)NC12CCC(CC1)C2)C C#Cc1ccccc1C(=O)NCC1(CNC(=O)C(CC2CC2)OC)CC1 N1(C(CC2(OC)CCOCC2)=O)CCC(O)(C(C)NC(C2CCCC2O)=O)CC1 c1(C(N(CCOCCN(C(C(CC)OC)=O)C)C)=O)ncc(OC)cc1F.C1(S)CC1 c1(C(=O)NC2CN(C(c3ccnnc3)=O)CC3(CC3)C2)cnc2ncccc2c1 O=C(C(C1=NOCC1)N1CCCC1C1CCCOC1)NC1CC1c1ccc(Cl)cc1 C(=O)(N1CCC(C(=O)NC(c2cnn(C)c2)C)O1)c1c(CC)ocn1 C(=O)(C(CNC(=O)C(C)OCC(C)C)CC(C)C)NCCN1CC(OC)C1.C(CO)S CCC(C)(C(=O)N1C2CCC1CC(CNC(=O)C(=O)NCC(F)F)C2)C(N)=O CC(C)C(C)(CNC(C1(C(C)(C)C)CCCC1)=O)NC(=O)CCc1ccon1 c1(CC(=O)NCC2C(C(C)NC(c3cnccn3)=O)OCC2)cccnc1O c1(C(N2C(CC(=O)N(C)CC3COCCO3)CC2)=O)ccnnc1O CCCCCCCCC(=O)NC1CN(C(c2cc3c(nc2O)CCCC3)=O)C1 CCC(C)C(O)C(C)C(=O)NC(CC(F)F)C(N1CCC2(CCCC2)C1)=O C1(C(N2CCC(CN(C(=O)C(C)(C)n3ccnn3)C)C2)=O)CCCC(C)(C)CC1 C=CCCCCNC(=O)C(C)(C1CCC1)NC(=O)C(C)NC(N)=O N1(C(=O)CC2SCCCS2)CCC2(CCCN2C(=O)CC2CSC2)C1 c1(C(=O)NC(C(=O)NC(c2nnc(O)n2C)C)C2CCOC2)ccnnc1O c1(CC(C(C)C)NC(C2C(c3n(CC)ccn3)OCCC2)=O)ccccc1Br C12(CNC(C3(CC)CC3(F)F)=O)CC1CN(C(C1(O)CCCCC1)=O)C2 C1(NC(c2cnc(CC)[nH]2)=O)CCC(CNC(=O)C(C2CC=CCC2)OC)CC1 c1(C(=O)NCC(=O)NCC(c2n(C)ncc2)O)sc2c(c1C#N)CCC2 C1(CNC(c2cc(CCC)on2)=O)CCN(C(C2CC(C)C2)=O)CC1(F)F c1(C(N(CC(CNC(c2nccc(C)n2)=O)C)C)=O)cc(N)c(C)cc1C N(C1CCC(NC(=O)CCCn2cc(-c3cccs3)nn2)c2ccccc21)C(C)=O n1(CCOC)cc(C(=O)NCCC2CCCN2C(C2CC(SC)C2)=O)nn1 N1(C(C2(OC)CC(C)C2)=O)CCC(F)(F)C(CNC(c2nc(Cl)sc2Cl)=O)C1 N1(C(Cc2c(C)ccs2)=O)CC(C)CCC1CNC(c1ccc(NC=O)cc1)=O N1(C(C2C(=C)C2)=O)CC2CCC1CN2C(C1(C#N)CCOC1)=O n1(CC(=O)N(C(CCNC(C2N(CCC)CCC2)=O)C)C)cc(C#N)cn1 C(=O)(C(CC1CCC1)NC(=O)C(C)(C)NC(C1CNC(=O)O1)=O)OC Nc1ccc2nc(-c3ccc(CN(C4CCCCC4)CCCO)o3)sc2c1 CC1(C)CC(NC(C2CSC2)=O)CCN(c2nnc(C#N)s2)C1 C(c1ccc2ncccc2c1)=CC(=O)NC1(CO)CN(C(c2ccc[nH]2)=O)C1 Cc1cc(C(C(=O)NCc2ccco2)N(C)C(C2(O)CCOCC2)C)cc(F)c1 c1(C(=O)NCCC2C(C)CN(C(c3ccon3)=O)C2)cc2scnc2[nH]1 C#CCC(C(=O)NC(C)CN(C)C(c1ccnc(N(C)C)c1)=O)C1CC1 C1(NC(c2nc(CC)oc2C)=O)CC2CC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 CN=c1[nH]c(=NCc2ccnc(OC(C)(C)C)c2)[nH]c(=NCC(C)CC(F)(F)F)[nH]1 N1(C(C2N(S(C)(=O)=O)CC2)=O)CC2CCN(C(c3cccc(=O)o3)=O)CC2C1 CCCCC(C)CCC(=O)NCCOCCNC(=O)CCc1ccccc1 N1(CC2CC(C)OCC2)C(=O)CN(Cc2ccccc2C(F)F)C1=O C1(NC(C2CC3(CC(C=C)C3)C2)=O)CC2CN(C(C3(C)CCOCC3)=O)CC2C1 c1(C(=O)NCc2nc(CC(=O)OCC)on2)cnn(CC)c1C1CCCC1 c1(NC(C(n2ncc(C)c2)C)=O)ccc(C(N)=O)cc1 C1(C(=O)OCC)(CC)CCCN1C(C12CC(CCO1)C2)=O CCCC(CNC(=O)Cc1ccsc1C)C(=O)NCC(=O)NC.OCC C(=O)(C(CC(F)F)c1ccccc1)NCC(C)(C1CC1)NC(c1cc(C)ns1)=O c1(C(=O)NC2C(NC(c3cccc(C(C)C)c3)=O)C2)cccc2c1CNC2=O N1(C(C(CC)C)=O)CCCOC(CNC(c2cnc(CO)nc2C)=O)C1 C1(CNC(C(CN(CC)CC)F)=O)CN(C(c2cccc(N)n2)=O)CC(C)(C)C1 N1(C(C(CN(C)C)O)=O)CC(C(=O)N(CC(C)(C)O)C)CC1CO C1(C(=O)NC2(CNC3CCCO3)CCC2)OCCCC1c1ccccc1 c1(OC)cc(C(=O)NCC2CCN2C(=O)CN2CCN(CC)CC2)cc(N)c1O C1(NC(C(CC#C)(C)C)=O)CN(C(c2cn(C3CC3)nn2)=O)CC(C)(C)C1 C1(C(=O)NCCC2CCCN2C(=O)Cc2cn[nH]c2)CC2C=CC1O2 C1(NC(C2CCC(=O)O2)=O)CCCN(C(C23CC2CNC3=O)=O)C1 Cc1ccncc1CC(N1CC(OCCNC(=O)CC2CC=CCC2)C1)=O C(CN=c1ccn2nccc2[nH]1)N(C(=O)CC(C)(C)C(F)F)C c1(NC(=O)NCCCC(C)(C)NC(C(OC)OC)=O)ccc(O)c(=O)cc1 c1(C(N(C2CCN(C(Cc3cc(CC)on3)=O)CC2)C)=O)ncnc(CC)c1F Cc1cc(O)c(Cl)cc1C(=O)NC1CCC(NC(=O)CSCCC(C)C)C1 Cc1ccnc(NC(C)(CCCO)c2nnnn2CC2CC2c2ccccc2)n1 C1(C(C)NC(=O)C2CC2)CCCCN1C(c1cn(C2CCOCC2)nn1)=O c1(C(N2CCC(CNC(CN(C(COC)=O)C)=O)C2)=O)c(C)oc2ccccc12 Cc1[nH]nc2c1CCC(C(=O)NCC1CCN(C(C3(C)COCCO3)=O)CC1)C2 C1(CNCC(OCC)OC)CC(C)N(CC(F)(F)F)C1 C1(CCC)CN(C(C2(C)CC2)=O)CCN1C(c1cc(C2CCCC2)nn1C)=O C1(NC(C(c2cn(C)nc2)=O)=O)CCCC(NC(=O)COC2CC=CC2)CC1 C1(O)(CNC(C2C(C(=O)OC)C2)=O)CCCN(C(C2(OC)CCC2)=O)C1 CC1CC(NC(=O)CCCC(N)=O)CN(C(c2ccc(C(F)(F)F)nn2)=O)C1 CC1CN(C(c2ccns2)=O)CC(CCNC(c2cc(C3CC3)ncn2)=O)O1 C1(C(C)NC(=O)Cc2ccns2)CCN(C(=O)CCC2CCC2)C1 N1(C2CCN(C3CCC(=O)NC3)C2)CCN(CC(F)(F)F)C(=O)C1 Cc1cc(CCC(=O)NCC(C)CNC(C2(C)CC(C)C2)=O)on1 C1(NC(C(c2ccc(Cl)cc2F)C)=O)CC2CCC1N2C(C1CCOC1)=O C1(CCNC(C(C)Cn2ccnc2)=O)CN(C(c2c[nH]c(=N)s2)=O)CCO1 c1(C(N(CCCN(C(C(CC)n2ccnc2)=O)C)C)=O)c(F)cc(F)cc1F c1(C(=O)NCC2(F)CC(NC(C3(C#C)CCC3)=O)C2)c(C)c(C)c(C)c(C)c1C C(=O)(C(CC(C)(C)C)C1CCOCC1)OCC(C)(C)OCC(=O)OC c1(CC)nnc(C)cc1C(=O)NCC1CCC(CNC(C2CCCSC2)=O)CC1 C(CCCCCNC(=O)C(C1CCCCC1)O)NC(=O)COCCF c1(C(=O)NCCC2CCCN(CC(N)=O)C2)ncccc1Cl C12CN(CCS1(=O)=O)C(=O)COCC2.c1(CC2C(C(=O)OCC)C2)ccnn1C N1(C(c2cnn(C)c2Cl)=O)CC(NC(c2nnc(S)n2C)=O)CC1(C)C N1(C(C(CNC(C=CCOC)=O)C)=O)CCOC(C2(O)COC2)C1 C(=O)(CCCCCn1cc(CONC(=O)OC(C)(C)C)nn1)NCCCCCC N1(C(CC2N(C(Cc3c(C)ocn3)=O)CCC2)=O)CCCC(OC2CC2)C1 c1(C(=O)NCC2CC(NC(c3cocc3Br)=O)C2)cccc(F)c1O n1(CC(=O)NC2CC(CO)N(C(C3COCCO3)=O)C2)c(O)nnc1O N1(C(COCCC)=O)CCN(C(=O)Cc2cccc(Br)c2C)CC1CO N1(C(CCC2CCN(C(CNC(CC)=O)=O)C2)=O)CC2(COC(C)C2)C1 C(C(C)(O)CC(=O)NC(C1CN(C(C2CC3(C2)CC32CC2)=O)C1)C)OC C(=O)(C#CC1CCC1)NCC1CC(C(=O)NC2(C)CC(N)C2)C1.C(C)(C)(C)O Cc1ccoc1C(N1CCCC1CN(C(=O)CNC(=O)CC1CCCCC1)CC)=O N1(C(CCN(CC)CC)=O)CCC2(CC2)CC1C(=O)NC(c1cncn1C)CO Cc1cc(F)c(Cl)cc1C(=O)NC1(C)CCC(NC(=O)C2=CCCOCC2)CC1 C1(C(=O)NCC(C)(C2CCC2)NC(c2nn(CC)c(C)c2)=O)COC(C)(C)CO1 CC1COCCN(C(=O)CS(N)(=O)=O)C1C C(=O)(CCC(=O)c1ccc(Br)cc1)NC(CNC(=O)C(F)=CCCF)CO C(C(=O)NC1CC(F)(F)C1)(C1=CCSC1(C)C)N(CC(N1CCCC1)=O)CC n1(CCOCC)ncc(I)c1NC(=O)Nc1cccc(OC)c1 C1(CC(=O)NCC2CCN(C(c3c(C)nc[nH]3)=O)C2(C)C)CCCCCC1(F)F C(=O)(C(C)C(O)C(C)C)NCCCC1(NC(c2cc(CC)ncc2)=O)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)N1C(CCNC(CCCCC)=O)CC(OC)C1 c1(C(=O)NCC(C)CN(C(=O)C(O)C2CCC2)C)cccc(C(C)(C)C)n1 c12ccccc1CC(=O)NC2.C1(C(COC)NC(=O)C(C)N2CCCC2)CCCC1 C1(CNC(C2(SC)CCC2)=O)CC2(CC2)CN1C(C1CCCC(CF)C1)=O c1(CN2CC3C(C(=O)Nc4c(CO)ccc(OC)c4)(C3)C2)c(Br)cc(Br)cc1Br C1(C(=O)NCC2(CO)CCCC2)CC2CC2N1C(=O)Cc1cnns1 c1(CN2C(C)(C(=O)Nc3cc(C(=O)OC)nn3C)CCC2)cc(Br)cc(Br)c1F CCC(C(=O)NC1(CC)CCN(C(C2CCCC(C)(C)C2)=O)CC1)C(C)C c1(C(N2C(C)(C(=O)Nc3ccnc(O)c3)CCC2)=O)cnn2cccc(F)c12 CN1CC2CN(Cc3cn(-c4ccnc(F)c4)nn3)CCN2C1=O N1(CCN(C2CCSC2)C(=O)Nc2cnn(CCF)c2)CCOCC(CO)C1 C1(C)(C(C)(C)C)CCCN1Cc1ccccc1C.CC c1(-c2c(C)ccc(CO)c2)cc(C(N2CC(C)(OC(C)C)C2)=O)c2cc[nH]c2c1 c1(C(=O)NC2C(NC(c3ccc(C)nc3O)=O)CCC2)ccc2c(c1)NC(=O)C2 N=c1ccc(C(N2CC3C(NC(c4csc(-c5ccoc5)n4)=O)C3C2)=O)n[nH]1 C1(CNC(C2N(C(CC(=O)OC)=O)CC2)=O)CC(C)OC(C)C1 C1(CC)CN(C(=O)Cc2ccsc2)CCC1NC(C1(N(C)C)CCCSC1)=O C12CC3CCC(C1)N3Cc1ccccc1N2.c1(NCC)c[nH]c(C)c1C(=O)OC C1(C)(NC(C2(CC)COC2)=O)CC(NC(=O)CCC2CCCN2C)C1 CCN=c1[nH]c(C(N2CCOC(CN(C(C3CNC(=O)O3)=O)CC)C2)=O)cs1 N1(C(C(C2CCOC2)OC)=O)CC23CCCC2(C1)CN(C(=O)CCP(C)(C)=O)C3 c1(CC)ccnc(F)c1Cl.CCCC1C(=O)N1.C12CN(CCS1)C2 c1(NC(C2C(NC(C(C#C)(C)C)=O)C2)=O)cc(C#N)ccc1Cl C(CCC(=O)NCc1nc(Cl)oc1C)(C(C)C)NC(C(CSC)OC)=O C1(C(=O)NC2C(CNC(=O)C=Cc3cncc(F)c3)CC2)CCn2nncc2C1 CC(CCCC(=O)Nc1ccc(O)cc1)NC(=O)C(C)(Cl)Cl c1(CNCC23C(CN(C(c4n[nH]c(C)c4C)=O)C2)C3)cccc(F)c1C#N c1(CC(C)C(N2C(C(=O)NCc3cccc(Cl)n3)CC3CC23)=O)ccc(O)cc1 c1(CN2CCC(CO)CC2C(F)(F)F)c(F)ccc(Cl)c1Br N1(C(C(Cc2ncn(C)c2)O)=O)CCC(NC(c2occ3c2CCC3)=O)C(O)C1 C1(O)(CC(=O)NCCC2CCCN(C(CC3CCC(C)C3)=O)C2)COC(C)(C)C1 c1(CN(CC)Cc2ccccc2Cl)nc(-c2ccc(Br)o2)oc1C C1(NC(C2(CNC(C3CCC(=O)O3)=O)CCC2)=O)C(CC2CC2)CCC12CCC2 c1(OC)nc(C(=O)NCCC2CCCN(C(C3(SC)CC3)=O)CC2)cc(O)n1 C1(c2ccccc2)CC2(CC2)C1.N1(C(C(=O)NCCc2ccccc2)=O)CCC(S)C1 c1(C(CNC(N(CC#CC)C)=O)C(=O)OC)ccc([N+](=O)[O-])cc1 Cc1nccc(F)c1C(=O)OC(=O)CCCCOc1ccccc1Cl N1(C(CCC(=C)Cl)=O)CCN(C(c2cn3c(n2)SCC3)=O)CC1C Cc1oc(=O)oc1S(=O)(=O)Oc1ccc2snnc2c1 CC1SCCCC1C(=O)NCC1CC(C(N2CC(F)C2)=O)CO1 c1(C(=O)NC2CCN(C(c3n(CC)nc(C)c3)=O)C2)c(Cl)ccc(Cl)c1F C1(CC(N2CC(O)(C(C(=O)N(CC=C)CCO)F)C2)=O)CCOC1(C)C N1(C(CSc2cccc(C)c2)=O)CCN(C(c2sc(F)cc2C)=O)C2CC12 c1(C(=O)NCC(C(=O)NC2COCC2CO)N(C)C)ccc2c(c1)CC2 N1(C(CN2CCC(C)CC2)=O)CC(C)(C)OC2(C1)CN(C(C1OCC1(C)C)=O)C2 c1(NC(C)=O)ccnc(C(=O)N(c2ccccc2)Cc2scnc2C)c1 C1(C(=O)NCc2cc(C)[nH]n2)CC(C)CN(C(c2occ3c2CCC3)=O)C1 CN1C(=O)CCCC1C(=O)N1CCC(C(=O)NC2(C3CC3)CCOC2)O1 N1(C(c2c(CC)nns2)=O)CC(CO)C2(C1)CN(C(c1ccc(OC)o1)=O)C2 N1(C(C2(OC)CCSC2)=O)C2CCCC1CC(NC(=O)CSc1n[nH]c(C)n1)C2 S(=O)(=O)(c1ccc(NCC23CCCC2C3(F)F)c(F)c1)N(CCC)CC N1(C(CC2C(CC)C2)=O)CC2CC1C2NC(c1cnn(C2CCOCC2)c1)=O c1(C(N(C)CCN(C)C(c2cnc(C(C)(C)C)s2)=O)=O)cc(Cl)ccc1C(F)F N1(CCc2cn(C(C(=O)NCC(C)C(=O)O)C)nn2)Cc2ccccc2C1 C(=O)(NN1CCCCC1=O)c1c(NC(=O)NC2CCCS2)cccc1 C1(C)(CNC(C(COC)N(C)C)=O)CCCN1C(=O)Cc1cnn(C2CC2)c1 c1(NC(c2ccc(F)cc2)CC(C)C)ncccc1S(=O)(=O)NCC1CSC1 N1(C(c2c[nH]c(=N)o2)=O)CCC2C(C1)CN2C(=O)CSc1ccccn1 c1(C(=O)NC2CCN(C(c3[nH]cc(C)c3)=O)CC2C(C)C)cc(C)c(N)cc1Cl C=C(C)CCCC(=O)N1CC(O)(C2CCCN2C(c2cc(C)c(Br)cn2)=O)C1 c1(CC(=O)NCCC2(O)CN(C(CCC(=O)NCCC)=O)C2)ccc(C)cc1F c1(C(=O)NCC=CCNC(c2ccc(C(=O)NC(C)C)cc2)=O)cnn2c1OCC2 c1(-c2c(F)ncc(SC)c2)ccc2[nH]c(C(N3CCOC4(CC4)C3)=O)nc2c1 CC(CN(C)C)CCC(=O)NC1(CO)CCCN(C(c2cccc(Cl)c2)=O)C1 c1(C(=O)N=c2cc[nH]cc2N2CCCC2)cnc2cccc(Br)c2c1 C1(NC(c2c(CC)nccc2)=O)CC2CC1CN(C(c1cnc(C)s1)=O)C2 c1(C(=O)OCc2scc(C(=O)OCC)n2)cn(C)nc1I C(CC(=O)NCC1(Cn2cc(CC(O)C3CC3)nn2)COC1)(OCC)OC C1(C(=O)NC2C(C)CN(C(C3CCOCC3)=O)C2)CCn2ccnc2C1 Cc1ccc2cc(C(=O)NC(C3(O)CN(C(c4cc(=O)cc[nH]4)=O)C3)C)[nH]c2c1 C(=O)(CC(C)(C)CC(=O)NCC(C)CNC(c1ccc(C(C)C)cc1C)=O)OC C(=O)(C(F)C1=CCCCC1)NCC1CCN(C(C2CCCCN(C)C2=O)=O)C1 c1(C(=O)NCC2C(NC(COCCC=C)=O)COC2)cc(N)ccc1F C1(C(=O)NC2C(SC)CN(C(c3coc(SC)c3)=O)C2)COc2ccccc2C1 c1(NCCN(C(c2c(C)c[nH]c2CC(N)=O)=O)C)nc[nH]c2nccc1-2 C(=O)(C1CCc2ccccc21)N(C(C(=O)NC(CSC)(C)C)C)C C(C(=O)N1CC(O)(CN(C(=O)COCCN(C)C)C)C1)(C(C)C)SCC N1(C(c2c(C)oc(CO)c2)=O)CCCN(C(=O)CCC(CF)CF)CC1C N1(C(C(CC)OC2CCCCC2)=O)CC(C)(C)CC1CNC(=O)CCOC(C)=O C1(CNC(C2CN(C3COC3)C2)=O)CCN(C(=O)CC2CCCCO2)CC1 C1(CNC(CC(CSC)(C)C)=O)CN(C(=O)C(C(C)C)SC)CC2(CCC2)O1 C1(CNC(C2C(CC)C2)=O)CCCN(C(C2CC2c2cccnc2)=O)C1 N=c1[nH]c2c(s1)CCCC2C(=O)N1CCC(CCNc2ncc(Cl)cn2)C1 c1(CNC(C2C(CNC(c3cc(CC)on3)=O)CCC2)=O)ccc(CO)nc1 c1(OC)cncc(C(N2CCOC(CNC(=O)CCc3ccc(Cl)cc3)C2)=O)n1 N1(C(C2OCC(C)(C)C2)=O)CCN(C(=O)C=Cc2cncc(F)c2)CC1C1CC1 c1(C(=O)NCC(=C)CCNC(C2CC2C(C)(C)C)=O)ccc(-c2cc[nH]n2)cc1 N1(C(c2cc(OC)cc(OC)c2N)=O)CC(NC(C2CC2C)=O)CC2(CCC2)C1 C1(NC(C(=O)Nc2c(F)cc(C)c(Br)c2)=O)CCOC2(CCSCC2)C1 N1(C(Cc2c(NC(C(CC(C)C)O)=O)cc(F)cc2)=O)CCC2(CC1)COC(=O)N2 c1(C(=O)NC)ccc([N+](=O)[O-])cc1C(N1CC2NCC1(C)C2)=O c1(C(C)C(=O)NCC2(NC(c3ccc(F)cc3)=O)CCOC2)nc(F)ccc1Cl O(CP(C)(C)=O)CC(=O)NC(C1CCCCC1)CNC(C1C(CCC)C1)=O c1(C(N(CCNC(c2scc(C(C)=O)c2)=O)C)=O)n[nH]c2c1CCCC2 c1(CC(C(N)=O)NC(C2C(NC(c3c(C)scc3)=O)CCC2)=O)ccc(O)cc1 C(=O)(C1=C(Cl)CCC1)NC(C(C)NC(=O)CN1CCC(N(C)C)CC1)CO N1(C(CCc2onc(CCC)n2)=O)CCC(NC(c2snnc2C)=O)C(F)C1 c1(NC(CSCC(=O)OC)=O)nc(C)cc(C)n1.C12CC1CNC(=O)CNC2=O C(=O)(C(C(C)(C)C)N(C)C)NCC1OCCN(C(CCc2nc(C)c(C)[nH]2)=O)C1 C1(C(N2C(CN(C(c3c(CCC)[nH]cc3)=O)C)COCC2)=O)CC(C)(C)CN1C c1(C(=O)NCC(CNC(CC(C=C)CC)=O)O)cc(Cl)c(C)cc1Br C1(N(C(c2cn(CC)nc2C2CC2)=O)C)CCCN(C(c2ccc(F)s2)=O)CC1 c1(OCC)cc(C(N2CC3CCCCCC3C2)=O)c([N+](=O)[O-])cc1OCC C12(C(=O)NCC(C(C)C)(C)NC(c3cc(C(F)F)ccn3)=O)CC1COC2(C)C c12nn(C)cc1C#CCCCC(C(=O)OC)CC1CCCN1C2=O C(=O)(C(C)(C)C(C)NC(=O)NCCOCc1ccc(Cl)cc1)OCC N1(C(C2CCN(CCC#C)CC2)=O)CCN(C(c2snnc2C)=O)CC(CO)C1 N1(C(C23N(C(c4cnn(C)c4C#N)=O)CCC2C3)=O)CCn2ncc(O)c2C1 N1(C(CC2(C=C)CCC2)=O)CCC(C)(NC(=O)C(c2ccccn2)C)C1 c1(CC(=O)NC23CC(NC(C=C4CCC(C)C4)=O)(C2)C3)ccc(F)cc1Br C(=O)(C1CCCc2ncccc21)NC1CN(C(C(CO)OC)=O)C2(C1)CCC2 c1(C(=O)NC2(C)CN(C(c3ccn4nccc4n3)=O)C2)cc(O)c2ccoc2c1 N1(C(C2N(C)C(=O)OC2)=O)CCS(=O)(=O)C(CCNC(c2ccc(O)nc2)=O)C1 CC(C)C(F)(CNC(C1C=CCS1)=O)C(=O)NCC1(c2ccon2)CC1 C1(CCC)CN(C(=O)CCCn2cncn2)CCN1C(=O)C(C)NC(=O)CC C(c1ccc(Br)cc1F)=C(C)C(=O)NC(C1CC(F)(F)C1)C Cc1ccc(C(C)CC(=O)NCC2(C)CCN(C(=O)C(F)(F)C3CC3)C2)cc1 C1(NC(c2nnc3n2CCCC3)C(C)C)CCCC(C2CCC2)C1 c1(CC)cc(C(=O)N(C(C)CNC(=O)CC2CCCCC2C)C)sc1C c1(C(=O)NCC2C(NC(C=C(CCC)C)=O)CC2)cc2c(C)ccc(Cl)c2[nH]1 c1(NC(c2c(NC(=O)CC3(O)CCOCC3)ccs2)=O)cc(Cl)cc2[nH]ncc12 N1(c2n(CCCOC)c(Cc3nc4cccnc4[nH]3)nn2)CCCC(C)(C)CC1 c1(CCCC(=O)NCCN(C(C2CCSCC2)=O)C2CC2)ccc(O)cc1 C(=O)(CCS(C)(=O)=O)NC1CC(N(C)C(c2n[nH]cc2Cl)=O)C1 C(=O)(C1OCCc2c(O)cccc21)N1CCC(NC(CCOC(C)C)=O)CC1C C=CCC(CNC(c1cn(C)c(C)n1)=O)C(=O)NC1CCCCNC1=O O=C(CCN=c1[nH]c(=NCCCF)[nH]c2c1CCC2)C1CCCC1 N1(C(C(C(C)O)C)=O)CCC(CO)(NC(=O)CC2OC(C)(C)OC2=O)CC1 Cc1nc(F)ccc1CNC(C1CCCC1NC(c1coc(Cl)n1)=O)=O C1(CNC(C(c2ccc(Cl)cc2)OC)=O)CCC(C)(C)CN1C(c1ccoc1)=O c1(N2CCC(COC)C2)nc(C)cc(=NC2CS(=O)(=O)C2)[nH]1 N1(C(c2c(SCC)nccn2)=O)CCC2C1CCCN2C(=O)CCC(C)(F)F N1(C(c2c(C)occ2)=O)CC(NC(=O)C=Cc2ccc[nH]2)C(C2CC2)C1 CC(C)(F)CCC(=O)NC1CC(C(F)C(N2CC(O)(c3nn[nH]n3)C2)=O)C1 N(C1CCOc2ccc(Br)cc21)S(=O)(=O)c1cccc(N2CCC3(CCC3)C2)n1 n1(C(C)(C)C)nccc1C(N1CCC(OCCNC(=O)Cc2csnn2)C1)=O C1(CNC(C(c2cccc(OC)c2)C)=O)C(C)CCCN1C(c1coc(Br)c1)=O C1(NC(CCC(C)(F)F)=O)CN(C(=O)CC2CCCCC23CC3)C2(CCCC2)C1 C1(CC(=O)NC(C(CO)NC(c2ccc(CC)o2)=O)C)CCCN(C(C)=O)C1 N1(C(C2CCN(C)CC2)=O)CC(C(N2CCC(CO)C(F)C2)=O)CC12CCC2 c1(C(C(N2CCCC(CNCC(CC)C3CC3)C2)=O)=O)cccc2c1OCC2 Cc1cc(C(=O)N(C2CCC(NC(c3ccnnc3C)=O)CC2)C)nc(C)c1 C(=O)(CC(F)(F)C(F)F)NCCC(C)N(C)C(C1C(F)(F)C12CC2)=O C12CC3(C1)CN(C3)CC(=O)NC2c1cnc[nH]1.CC(C)CC(C)N1CCCC1=O N1(C(C(C)C#N)=O)CCC(NC(C23CC2C3)=O)C(C)(C)C1 N1(CC(COC)NC2CC3C=CC2C3)CCN(C(=O)OC(C)(C)C)CC1 N1(C(c2ccc(F)cc2O)=O)CC2CCC1C(NC(c1ccc(CO)cc1)=O)C2 C(=O)(CCCCCC(C)O)N1CC(N(C(C(C(C)C)CC2CCCC2)=O)C)C1 CC(CN(C)C)CCC(=O)NCCCN(C)C(C1(F)CCN(C)CC1)=O C(=O)(CCC(C)N(C1CC(NC(c2ccc(SC(F)(F)F)s2)=O)C1)C)OC c1(C(N2C(CNC(CC=CCC)=O)CC2)=O)nnn(C2CC2)c1C c1(NC(C2C(NC(c3cccc([N+](=O)[O-])c3Br)=O)C2)=O)ccc2sc(Cl)nc2c1 Cc1csc2ncc(C(=O)N(CCNC(=O)C(F)n3cccn3)C3CC3)n12 CP(C)(=O)C1CCC(C(=O)OCc2cc(-c3ccco3)on2)C1 C(CCC(c1ccccc1)NC(=O)Cc1cnco1)NC(CSCC=C)=O C(C(=O)NCC1CC1)(C1CCSC1)N(C)CCC1(C)CC1 C=CCC(C)(C)C(=O)NCC1CN(C(=O)C(F)(F)CO)CC1O C1(C(C)C(=O)NC(C)C2CC2)CCCN(C(=O)C(C)(C)N(C)C)C1 C(=O)(CCCC(=O)NCC)NCCCC1OCCN(C(C(COCC)C)=O)C1 Cc1cc(C(=O)NC2CN(C(=O)Cc3cc[nH]c3)CC2F)c2cccc(C)c2n1 C1(C(N)=O)CCc2nc(NC(c3cc(Cl)c(F)cc3F)=O)sc2C1 CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)CC1NC(=O)C1=NNC(=O)C1 c1(OCCNC(Cc2cccc(CC(C)C)c2)=O)cc(Br)ccc1C#N N1(CC(=O)NC(C2(O)CN(C(=O)COC3CCOC3)C2)C)Cc2ccccc2C1=O CCCCS(=O)(=O)NCC(N1CCOC(CNC(=O)C(F)(F)CO)C1)=O C1(CNC(c2n(CC)ncn2)=O)CCC(C)N(C(c2cncs2)=O)C1 C1(N(C(C=CC)=O)C)CCCCN(C(C2CC=C(C)CC2)=O)C1 C1(CC)C(NC(=O)C=Cc2ncc[nH]2)CCN1C(C1CCS(=O)CC1)=O Cc1nc(=NC2CN(C(C3CC4CCC(C3)S4)=O)CC2C)s[nH]1 N1(C(C(CCC)C#N)=O)CCC2(CC1)CC2CNC(=O)Cn1cc(C)cn1 N1(C(CC2CC(C)(C)C2)=O)CC(F)(F)CC1CCNC(C1CCS1(=O)=O)=O N1(C(Cc2c(C)cccc2)=O)CC2(C1)CN(C(=O)N(CC(C)C)C(C)C)C2 C1(C(N2C(C(=O)NCCCCCC)C(O)CC2)=O)CCC2(CC1)CC2 Cc1ccc(C(N2CCC2(C)C(N2CCC(Br)CC2)=O)=O)cc1C(F)(F)F C1(N(C(c2ccc(N)cn2)=O)CC)CCCN(C(c2ccc(C)cc2)=O)CC1 C1(CNC(C2C(NC(c3nc(C)oc3)=O)CC=CC2)=O)CCC(C)(C)CC1 C1(C2CN(C(C34CCCN3CCC4)=O)C2)(NC(C(CC)N2CCCC2=O)=O)CC1 C12COCCC1C(=O)N2.C1(C(=O)NCc2cc(C(N)=O)co2)(OC)CCOC1 c1(C(N2CCCC(CC(=O)C3CC3)C2)=O)ccc2nc(-c3ccoc3)sc2c1 N1(C(C2(C#N)CC(C)C2)=O)CCC(NC(C2(C)CCCC2)=O)C(C)(C)C1 C1(CNC(CC2CCN(C(C34CC(CCC)(C3)C4)=O)C2)=O)CC(=O)N(CC)C1 C1(NC(=O)OC(C)(C)C)CN(C(=O)NCCc2cc(Cl)cc(Cl)c2)CC1C1CC1 C(=O)(CC(C(C)CC)NC(=O)CC1CSCCO1)Nc1ccc(COC)cc1 c1(OCC=C)ccc(C(=O)NC(C)C(C)NC(=O)CC2CCSCC2)cc1 c1(C(=O)NC(C(C)C)(C)CNC(C2CCCCCC2)=O)cnn2c(=O)cc[nH]c12 C(N=c1[nH]nc(C(N)=O)s1)C1CCCN(C(C2(C)C=CCCC2)=O)C1 N1(C(c2cn(CC)nc2C)=O)CCC(C2CCCN(C(=O)CCC(C)O)C2)CC1 Cc1ccc(NC(C2CC2[N+](=O)[O-])=O)cc1.C1(N)C=CCN1C(=O)CN1CCCC1 C1(C(=O)NCc2occ(C(N)=O)c2)CCCCC(=O)N1 C(=O)(N=c1ccn(CC(=O)N(C)C)[nH]1)C1C(C(C)C)OCC1 N1(CCC)CCC(CC)(NC(c2nn[nH]n2)=O)CC1 C1(O)(CNC(CCCc2scc(C)n2)=O)CCN(C(=O)CSC(F)(F)F)CC1 c1(NC(N2CC(=O)NC2=O)c2n(CCC)nnn2)ccc(-c2nnc(C)o2)nc1 S(=O)(=O)(C1CCOC1)NC(c1cc(C(C)C)nn1-c1ncccc1Cl)=O C1(CCOC)(C(=O)NC(c2cn[nH]c2)C)CCN(C(C2CCCCS2)=O)CC1 c1(OC)ccc2cc(C(N3CC(CNC(=O)C(C)(F)F)CC(C)C3)=O)nnc2c1 C=CCCC(C(=O)OC)NC(c1cc(OC)c(-c2cc(F)ncc2C)cn1)=O c1(SC(C(=O)N(C2CCN(C(CCNC(C)=O)=O)C2)C)C)ccc(C#N)cc1 N1(C(c2cc(C)[nH]c2)=O)CC2(CC2)CC1C(=O)NCCc1ccon1 CC1CC(CNc2cnn(C3CCCCCC3)c2)N(C(=O)OC(C)(C)C)C1 Cc1ccc2nc(-c3nc(CC4CCOCC4)nn3C(C)C3CC3)cn2c1 CC1CCC2(CCC2)CN1C(=O)NC1CC1(c1ccc(Br)cc1)C c1(OC)ncc(C(N2CCC(O)(CNC(c3ccc(Br)c(C)n3)=O)C2)=O)cc1C C1(CNC(C2(S(N)(=O)=O)CC2)C)CC2(C1)CC(F)C2 Cc1cnn(CC(=O)NC2CCC(CNC(C3CCOC3=O)=O)C2)c1 CCC(C)C(CC(=O)N(CC(C)OC)C)NC(=O)C(O)CC(N)=O n1(CC(N2C3CN(C(C(CC(C)C)F)=O)C(C3)C2)=O)ccc2ccc(F)cc12 C12CN(CC(C)(C)O1)C2.C1(NC(C2CC(N(C)C)C2)=O)CCN(CC(F)F)C1=O c1(OC)nccc(=NC(=O)C2CCN2C(c2cc(C)ccc2F)=O)[nH]1 N1(C(c2c(N)nccn2)=O)CCOC2CN(C(=O)COc3cnc(Cl)nc3)CC12 c1(C(=O)NCC2CCN2C(c2csc(-c3ccsc3)n2)=O)cccc(F)c1F Cc1nc(CC(C)C)c(C(=O)NC(C)C(CO)NC(=O)CSC(F)(F)F)s1 N1(C(c2c(C)ocn2)=O)CC2CCN(C(=O)Cc3ccccc3S(N)(=O)=O)CC12 n1(CC)ccnc1C(=O)NCCCCCN(C(=O)CC1CC1(Cl)Cl)C c1(C(=O)NC2C(CNC(CC(C)CF)=O)C2)c[nH]c2ccncc2c1=O C1(C(N(CCCNC(=O)C(C(C)C)n2cncn2)CC)=O)CCCC(C)(C)O1 C(CC1=CCN(C(c2csnc2Cl)=O)CC1)NC(c1c(OC)ccs1)=O C(=O)(CC(=O)NCC(CNC(=O)CC1CCCOC1)CO)OCC c1(OC)cccc(C(C)=CC(N2CCN(C(c3ccc(C)s3)=O)C(C)C2C)=O)c1 CN1CCC12CN(C(C13CC(CN1C(C1CCCCC1(C)C)=O)C3)=O)C2 N1(C(=O)NC2CCCC2Oc2ccccc2)CCNC(c2ccc(Br)cc2)C1 N1(C(C2CCC(C)(C)OC2)=O)CCCC12CCCN(C(=O)C=CC=C(Cl)Cl)C2 c1(C(N2C(C(N3CCN(S(C)(=O)=O)CC3)=O)CC(=C)C2)=O)ccc(Cl)c(OC)c1 N1(C(C(C)OCC)=O)CCC(NC(c2cnc(F)c(Cl)c2)=O)C(CC)C1 c1(C(=O)NCCC(C)NC(C2CCOC2C(F)(F)F)=O)ncc(C(F)F)s1 N1(C(CC=CC(=O)N(C)C)=O)C(CNC(C2CC2(C)C)=O)CC2CCCC12 CC1CN(C(=O)C#N)CCN1C(C1(c2cc(Br)ccc2O)CC1)=O C(CCF)(C(=O)N1CCN(c2ncco2)CC1)OCC(=O)NC1CC=CC1 c1(OC)ccnc(C(=O)NC(CNC(=O)C(O)CC(C)C)C(C)C)c1OC C(=O)(CCCS(N)(=O)=O)NCCC1N(C(CCC(C)c2c(C)ncs2)=O)CCSC1 N1(C(C2(OC)CCOCC2)=O)CCC(CC(=O)O)C(NC(c2[nH]cnc2C)=O)C1 N1(C(C)C)CC(NC(=O)CN(C)C(N)=O)CCC1=O.N12CC(C(C)C1)C2=O C1(NC(Cn2c(C)nnn2)=O)CN(C(c2ccc(C(C)C)c(F)c2)=O)CC1(C)C C(C(COC)C(=O)N1CC(N2CCN(C(C3(COC)CC3)=O)CC2)C1)OC c1(C(=O)NC(C)CN(C)C(C2CCC(=O)N2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NC(CSC)C)ccc(CNC(=O)CC2CC(C)=NO2)s1 c1(C(=O)NCC(C)(CO)NC(CC2(COC)CC2)=O)cccc2nc(C)nn12 c1(C(N(CCNC(c2cccc(CC)n2)=O)C)=O)ccc2c(c1)COCO2 Cc1ccc(Br)c(F)c1CNC1CCC(=O)NC1=O c1(C(=O)NC2CC(NC(c3c(COC)ncs3)=O)C2)cnn(CC(F)(F)F)c1C Cc1ccc(C)c(C(=O)NC2(CNC(=O)C3=CCSC3)CCC2)c1 c1(C(=O)NCC(C2CC2)NC(C2(OCC)CCOC2)=O)cnc(=NCCF)[nH]c1 C(C(C)(C)CN(C(=O)COCCOC)C)NC(C(C)N(CCC)C)=O N1(C(c2c(CC)ncnc2)=O)CC2CC(NC(C3(C4CCC4)CCC3)=O)CC2C1 C=CC(C(=O)NC1CCC1OC(N1CCCCC1)=O)NC(=O)OC(C)(C)C C12C(CCN1C(=O)CC1CCCN1C)CNC2=O.C1(=O)CN1.N(CC)(CC)CC N1(C(CCOCC#C)=O)C(C(=O)NCC2CCCSC2)CC2CCCC12 c1(CC(=O)NC2CCCN(C(c3c(SC)cn(C)n3)=O)C2)c(C)cc(C)cc1C c1(CC(=O)NC(C2CN(C(=O)CCN3CCOC3=O)C2)C)csc(S)n1 C1(C)(CNC(C(CC2CCCC2)NC(CCC)=O)=O)CC(C)(C)C1 Cc1ccc(C(=O)NC2CC(C(N3CC(OCC(N)=O)C3)=O)C23CCC3)nc1O CC(C)C1=CCC(C(=O)N(CC(=O)N(C)CC2(C)CCCO2)CC(C)C)CC1 c1(CC)oc(C)cc1C(=O)NCc1nnn(C)c1C(=O)NCC1CCCSC1 Cc1cn2ccc(C(=O)NC3COCC3NC(C3(Sn4cccn4)CC3)=O)cc2n1 c1(C(=O)NC(C)CCNC(c2c[nH]nc2C2CCCC2)=O)ccc(Cl)cc1O C(=O)(CCCC(=O)N(C)C)NC1CN(C(c2c[nH]c(=NC)o2)=O)C(C)C1 C(CCCN=C(NCC(NS(=O)(=O)NC)c1ccco1)NC1CCNC(=O)C1)SC O=C(C(F)C(F)(F)F)N1CCN(C(C2(NC(=O)C3CC3)CC3(CCC3)C2)=O)CC1 C#CCC(C)(C(=O)N1CCC1(C)C(=O)NCC=C)NC(=O)CC1CCOC1(C)C c1(C(=O)NC(CC=C)CNC(C2CN(C(C)=O)C2)=O)ccc2cc(Cl)ccc2c1 C(=O)(C(C(C)C)c1ccn(C)n1)N(CCCNC(COC(C)C)=O)C c1(C(=O)OCC)ccc(Br)cc1NC(=O)Nc1c(I)n[nH]c1C N1(C(C(c2cccc(Cl)c2)C)=O)CCC(NC(c2n[nH]cc2C2CC2)=O)C1C c1(CC(=O)NCC(O)CNC(c2ccc(C(F)F)nc2)=O)cncnc1O N1(C(CCNC(=O)NC)=O)CCC(F)(CNC(C2(C3CCCOC3)CC2)=O)C1 c1(OC)ncnc(OC)c1C(=O)NC1CCN(C(=O)CN2CSCC2=O)C(C)C1 c1(C(=O)NCC(c2ccccc2F)NC(CCC#C)=O)cnc2ccccn12 c1(C(=O)NCC(CC(C)C)NC(C2(C)CC=CCC2)=O)c(F)ccnc1Cl C(=O)(C#CC(C)(C)CNC(c1ccncc1Cl)=O)N1CCC(NC(C)=O)C1 Cc1cc(F)ccc1-c1csc(NC(=O)Nc2ccccc2CO)n1 CC(=O)CCC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cnsc1)C C1(CC(N2CC(NC(C3CCN(CC)C3)=O)C(C)C2)=O)OCCCC1(C)C c1(OC)cccc(C2CC(O)CN2C(=O)C(C)n2ccnc2)c1 N1(C(c2ccc(C#N)cc2)=O)CCC(C2CCCN(C(c3ccoc3Cl)=O)C2)C1 N1(C(c2cnc(CCCC)s2)=O)CCC(NC(c2cnn(CCC)c2Cl)=O)C1C C1(CN(C(=O)CSCCC#N)C)CCCN1C(=O)CCc1ccncc1 c1(OC)ccc(Cl)c(C(=O)NCCCN(C2CCCCC2)C(C2CCC=CO2)=O)n1 CC1C(C(=O)N2CCC3(CC3C(=O)NCc3cnc4n3CCC4)C2)=NOC1C Cc1cc(C(=O)NCC2CN(C(=O)C(c3ccn(C)n3)C)CC2O)cc(F)c1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NC(CC)CNC(C1C2CCCC12)=O N1(C(c2nn(CC)nc2C)=O)CCC(C)C(CNC(c2cc(F)cnc2Cl)=O)C1 C#CC1(C(=O)NC(C)C(C2CC2)OC)CCN(C(c2ccc(CC)o2)=O)CC1 C(C(C(=O)OC)N(C)C)N.n1(CC=C)cc(C(=O)NCC(O)C(=O)NC)nn1 C=C(C)CCC(=O)NCC(C)(C1CC1)NC(=O)CN1C(=O)C1.C(C)(C)(C)OC(C)=O C1(C(N2C(CNC(=O)Cc3csc(S)n3)CC(OC)C2)=O)CCc2ccnn2C1 N1(C(c2c(OC(C)C)cccn2)=O)CCN(C(=O)Cc2ccco2)C2CC12 c1(-n2cc(OC)nn2)cnn2c1OCCC2.c12cc(cc(SC)c1)C(=O)N2C1CC1 c1(CC(=O)NCC(CC)NC(=O)CC2CC3CC3C2)cnn2ccccc12 C1(NC(CCCc2onc(C)n2)=O)CC2CN(C(c3nc(Cl)oc3C)=O)CC12 C=C(CNC(=O)CSc1n[nH]c(C)n1)CCNC(=O)CC1(CO)CC1 C(C1=Cc2ccccc2OC1)=CC(=O)NC1CN(C(C2CCC(F)(F)CO2)=O)C1 C1(CC(=O)NC2C(CNC(c3c(CC)scn3)=O)CCCC2)CCC(=O)NC1=O C1(CN=C(NCC2(OC)CCC2)NCC(F)F)CCOC2(CCOC2)C1 c1(CC(=O)NC2C3CCN(C(C(C)SC(F)(F)F)=O)C32)ccnc(Cl)c1F N1(C(C(N)CCSC(F)(F)F)=O)CCCC(c2ccncc2)CC1 N1(CCC)CCC(C(=O)NC2CN(C(=O)CN(C)C(C)C)C3CC23)CC1 c1(CC)oc2ccccc2c1C(N1CCOC2(C1)CN(C(=O)C(C)(F)CC)C2)=O C#Cc1ccc(C(=O)NCC(CO)NC(=O)CN2CCCC2C)c(F)c1Cl CCCC(C(=O)OC)C(=O)N(CC(O)CNC(=O)COC(C)C)C N1(C(c2cnn(C)c2Cl)=O)CCC2(CCN(C(C3CCCCS3(=O)=O)=O)C2)C1 CCC(C)C(C(=O)NCC(C)S(N)(=O)=O)NC(c1cnn(CCF)c1)=O c1(CNC(c2cncc(NC(C3CCOCC3)=O)c2)=O)ccc(Br)c(F)c1 Cc1ocnc1CCNC(=O)C(c1ccnn1C)NC(=O)COC1CC=CC1 c1(CC(=O)NCC(CC)NC(c2nocc2Cl)=O)csc(C2CCOCC2)n1 C1(N(C(CNC(CC)=O)=O)C)CCCN(C(c2cc(Br)c[nH]2)=O)C1 Cc1cc(F)cnc1C(=O)N(C)CC1COCCN1C(c1cnc(C)c(C)c1)=O C#CCC(C)(C(=O)NC(CO)CC(C)CC)NC(c1nonc1C)=O CC1CN(C(=O)C(C)N(C)C)CCN1C(C1CCC(C)(C)OC1)=O C(C)(CCNC(=O)COCCN(C)C)N(C(C=C(CC)C)=O)C N1(C(C(C)S(N)(=O)=O)=O)CCC2C1CCCN2C(c1nccc2n[nH]cc12)=O C1(CNC(c2cc(OC)ns2)=O)N(C(=O)CN(C2CCSC2)C)CCCC1(C)C C(=O)(C1CCc2cc(Br)ccc21)N1CC2CN(C(C(C)C)=O)CC2(C)C1 CC1CC2CN(C(=O)C(C)c3ccco3)CC2N1C(=O)CCCC1CC1 O=C1CSC(C(N2CC=CC2C(N2CCC(n3ccnc3)C2)=O)=O)C1 Cc1cc(Cl)nc(Cl)c1C(=O)NC1CC1C(N1CCNC(=O)C1)=O CCC(C)(C(=O)O)N1CCN(C(c2cnns2)=O)CC1 Cc1nn(CCO)c(C)c1C(=O)NC1CCN(c2ccc(Cl)c(F)c2)C1 CC1(C)CN(C(=O)Cc2ccccc2O)CC1NC(=O)C(O)Cc1ccccc1 CC(C(=O)NC1CCN(C(=O)Cc2cc(C3CC3)nn2C)C12CC2)C(C)(C)C Cc1ccc(C(N2CC(CC(=O)NC3CC(C)OC3=O)C3(CC3)C2)=O)c(O)c1 Cc1nccc(C(N2CCCCC(C(=O)N(C)Cc3cncn3C)C2)=O)c1N N1(C(C(COC)C)=O)CC(OC)C(C(=O)N(C)Cc2ccccn2)C1 c1(C(N2Cc3cccnc3C2)C(=O)NCCCF)nc(Br)c2ccccn12 c1(C(N(C(CCNC(c2cc(CC)[nH]n2)=O)C)C)=O)ccc(C(C)=O)cc1 C(CC(=O)NCC(F)(F)F)N(CCOC)C.C(CCN(C(=O)COCC)C)OCCO N1(C(C2(OCC)CC2)=O)CCC(NC(=O)C(F)C2CCCC2)C1 c1(NC)cnncc1C(=O)NC(CN(C(C1C(CNC)CC1)=O)C)C c1(C(N(CC(C)NC(c2ccc(Cl)s2)=O)CC)=O)cncc2ncn(C)c12 c1(OC)c[nH]nc1C(=O)NC1CCN(C(C2CC(C(C)C)C2)=O)C1 c1(NCc2cn(CC(CNC3CCCCC3)OC)nn2)cc(Cl)n(C)n1 C(=O)(C(CNC(c1ccc(F)cc1)=O)CC1CCCC1)NCCNS(N)(=O)=O C1(CSC)CCC2CCCCC2C1.C12(CC1)C(=O)N(C)CCN(C)C2=O c1(C(=O)NC2CCCCN(C(=O)CN3CC4CCC3C4)C2)cnc2nccn2c1 C1(CC(=O)NCC(C)(C2CC2)NC(c2cc(OC)n[nH]2)=O)CCCCN1C c1(C(=O)NCCOCCCNC(c2c(CC)noc2)=O)[nH]cc2c1CCCC2 N1(C(CC2CCC(C)(C)C2)=O)CC2(CC2)CC1CNC(C1CC=CCC1)=O CCC(CC(=O)NC(C)(C)C(C)NC(=O)C=C(C)c1ccco1)c1ccccc1 C1(C(=O)NCC(C)CNC(=O)CCc2cn[nH]c2)C2CCN(C)CC12 c1(OCC(N2C(CNC(C(C)OC)=O)C3CC3C2)=O)cccc(F)c1F c1(N(C)CC)ccccc1-c1cnc(-c2ccccn2)s1 N1(C(c2cnc(CC)nc2)=O)CCC=C(CNC(=O)CC(C)(C)CN(C)C)C1 c1(OC)cccc(C(=O)NC2CN(C(c3csc(F)c3)=O)CC2C(F)F)n1 C1(C(=O)NC(C)CNC(=O)CCc2cnco2)CCC(=O)N1 CC1(C)CC(NC(C2(C)CCC(=O)N2)=O)CN1C(C12CC(F)(C1)C2)=O C1(C(N2CC3C(CNC(c4cc(O)nc(O)c4)=O)C3C2)=O)CCCCC12CCC2 N1(C(c2c(C3(C)CC3)c[nH]c2)=O)CC(C)(C)C(NC(=O)C(Cl)=CCl)C(C)(C)C1 C(=O)(C(CNC(=O)CCn1ccnc1)CC1CC1(Cl)Cl)NCC(C#C)OC N1(C(C2CC(SC)C2)=O)CCCC(C)(C)C1CNC(c1cncn1C)=O C1(CC(=O)NCCOC(CNC(c2n(C)nnc2)=O)(C)C)CCC(C)(C)O1 CN=S(=O)(c1ccc(C(=O)NCC2CCC(NC(=O)N(C)C)CC2)cc1)N(C)C Cc1cccc(F)c1C(=O)NC1CN(C(=O)CCc2cnoc2)CC1C(F)F c1(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)C(F)(F)F)cccc2c1COC2 c1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)N(C)C)C2)n[nH]c2c1CC1CC21 O=S(=O)(c1csc2ccc(Cl)cc12)NCC1COCCC1(F)F CC1CCN(C(c2ccc(CO)cc2F)C(=O)NCc2cnn(C)c2)CC1(F)F Cc1ccc(CC(N2CCC(NC(c3cc4sc(C)cc4[nH]3)=O)C2)=O)c(F)c1F c1(C(N(CCC(C)(C)NC(C2C(c3n(C)ncc3)C2)=O)C2CC2)=O)cncc(N)n1 C1(CNC(C(CC#C)C2CC2)=O)CCN(C(=O)CCCCC)CCC1(F)F C(=O)(CC1=CCCCC1)NCCCCCN(C)C(C1(C)COC(=O)C1)=O n1(CC(N2C(CNC(CSCC(C)C)=O)C=CC2)=O)nc(C2CC2)n(C)c1=O c1(C(N2CC3CC(O)CC2C3)=O)cc(Br)c2nccn2c1 N1(CC(=O)NC(CNC(C(C)SCCCC)=O)C)C(=O)CCCC1=O N1(C(C2C(C(C)C)CCO2)=O)CCCCC1CC(=O)NC1(C)CC1C CCC(C)C(C(=O)N1CCCC1CCCO)N(C)C(C1OCCC1CN(C)C)=O N1(C(c2cc3cc(CC)sc3s2)C(=O)NCC)Cc2ccc(OC)cc2CC1C c1(C(N(CCC(C)NC(C(CC)OC)=O)C)=O)cc2cc(F)cc(F)c2[nH]1 N1(C(c2cccc(C)n2)=O)C2CCC1CC(NC(C13CCC1C3)=O)C2 c1(C(N2C(CN(C)C(c3nnsc3N)=O)CCC2)=O)ccc(O)nn1 C1(NC(c2cccnn2)=O)CCCC12CN(C(c1cc3nc[nH]c3cn1)=O)C2 C1(CNC(c2c(C)cns2)=O)CCCC(NC(=O)Cn2ncnn2)C1 C1(CC)CCC(N=c2ccnc(N3CCCN(C(c4cc(Br)cs4)=O)CC3)[nH]2)C1 C(c1nc2ccccc2[nH]1)=CC(N1C(CNC(C(C(C)C)(C)O)=O)CC(F)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(CC(C)O)=O)CC(F)(F)F Cc1cn2c(C(C3CCCC3)NC3CN(C(=O)C(C)CC(N)=O)C3)cnc2s1 c1(C(N2CCC(C(C)C(=O)NCC3(C4CCC4)CC3)C2)=O)ccnc2cc[nH]c12 C1(C(C)C)CN2CCCC2CN1C(=O)NC1CC(=O)C12CCC2 c1(C(=O)NC2C(NC(CCCC)=O)CCC2)ccc(C(C)C)cn1 c1(OC)cccc2ccc(C(=O)NCC(C)NC(c3cc(=O)n(C)cn3)=O)nc12 CC1CN(C(=O)CCc2nncs2)CC1(C)CNC(=O)C(c1cccn1C)=O C1(NC(=O)COC2CCOC2)(CO)CN(C(C2CC2c2ccncc2)=O)C1 C1(C(=O)NCCNC(c2cncc(C#C)c2)=O)CC2(CCOCC2)CO1 N1(C(C2(C)CC(=O)C2)=O)CCC2(C1)c1[nH]cnc1CCN2C(c1sccc1F)=O O=S(=O)(c1[nH]c(=NCC2CSCCO2)ccc1Br)N1CC=CC1CF C(CC(CC)C(=O)N(CCCNC(=O)CC(C(F)F)c1ccc(F)cc1)C)=CC C1(C(=O)OC(C)(C)C)CCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 Cc1cc(CNC(=O)C(C)N(C(c2cc(F)n(C)n2)=O)C2CC2)cnc1F C1(C(N2C(C(=O)NC3CC(C)(CC)C3)C3CC3C2)=O)CC2OC1C1CC21 c1(C(=O)NCC2(NC(c3cnn(C(F)(F)F)c3)=O)CCC2)ccc2c(c1)CCO2 N1(C(c2ncn(C)n2)=O)CC2(CC(CNC(c3cnn(C4CCC4)c3)=O)C2)C1 C(=O)(C1=CC(C)(C)C1)NCCC(CNC(=O)CC1(C)CCCO1)OC C(CCC(=O)NCc1cn(C2(C(=O)OC)CC2)nn1)NC(N)=O CCCC(O)CC(=O)NCCCCN(C(c1scnc1C1CC1)=O)CC N1(CCC(=O)NCC(CN(C(c2c(C)nsc2)=O)C)C)CCCCCC1 N1(C(C(n2cc(CN3CCCC3=O)nn2)C)=O)CCC(O)C(C)(CO)C1 Cn1cc(C#N)cc1C(N1CCC(O)(CNC(=O)CCC2CC2(F)F)C1)=O c1(CN2C(C(=O)Nc3cnc(C(=O)OCC)nc3)CC3CC32)cc2cn[nH]c2cn1 C(=O)(C(CC(C)C)NC(=O)Nc1sc(C)cc1C)NC(CC#C)(C)C N1(C(C2N(C)CC2)=O)CCCC2(CCCN2C(C2CCc3c[nH]nc3C2)=O)C1 c1(CC(C)C(=O)NCC2CC2CNC(c2cnc[nH]2)=O)ccccc1.C(C)(C)C CC(C(=O)N1CCCCC(NC(c2ccsc2C#N)=O)C1)C(F)(F)C(F)F c1(C(=O)NCC2OCCC(NC(C3C(OC)C3)=O)C2)cc2c(Cl)nccc2o1 C1(CC(N)=O)(NC(C(CC#C)O)=O)CCN(C(=O)C(C)(CC)OC)CC1 C1(n2c(C(CC)O)nc(CC(C)CC)n2)CC2(C1)CC1(CCCC1)C2 CC1(C)CCN(C(C2CCCCS2)=O)C1CNC(c1cccc(F)c1F)=O c1(C(=O)O)ccc2c(c1)CC(C(=O)O)CN2CC(c1ccc(Cl)cc1)(F)F c1(CNC(c2cscc2Cl)=O)ccccc1COC(c1ncncc1Cl)=O C(C1=CCN(C(=O)CC2(C(F)F)CC2)CC1)NC(C(C(C)C)NC=O)=O O=C1CC2CCC1C(NC(=O)N(CCC1CC1)CC1CC1)C2 C(=O)(CCCCC(=O)NCC1CC1NC(=O)COCCc1cccs1)OC c1(OC(C(=O)NCC(C)NC(C(CC)N2CCCC2=O)=O)C)cccc(C#N)c1 COn1cnc(C)c1C(=O)NCc1cc(C(=O)NCC(C)CCCO)ccn1 N1(C(C=COCC)=O)CCC2C(CCN2C(C2C(C(=O)OC)C2(F)F)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC(C)CN(C)C(C1CCCCN1S(C)(=O)=O)=O C1(NC(=O)Cc2ccccc2)CCN(C(C2CCCC23CC3)=O)CC1 N1(C(c2ccccn2)=O)CCN(CC2CN(C(c3scnc3Cl)=O)C2)CC1 Cc1cnc(N2CCOC(CN(C)C(c3cc(Cl)nn3C)=O)C2)nc1 c1(OC)ccc(C(=O)NCCC(C)CCNC(c2cc(SC)oc2C)=O)c(F)c1 C(C(C)(C)CNC(c1ccoc1Cl)=O)N(C(C1C(CC)C1)=O)CC Cc1nc(Cl)ccc1CC(=O)NCC1CCCCC1NC(=O)C(C)n1cccn1 N1(C(=O)OCC)CC2CCC1C(C(C)NC(=O)C(C)CNC(=O)C(C)(C)F)C2 C1(n2cc(CC3CCNC3)nn2)CCC(=O)NC1.CC(C)(S(C)(=O)=O)C1CCOC1 C1(C(C)C)CN(C(=O)CCn2cc(-c3cc(C(=O)O)ccc3Cl)nn2)CC(=O)N1 C(=O)(CCC(CC)CC)N1CCC2(C(N(CCCC)CCCC)C2)C1 N1(C(=O)NC2CCCN(CCS(C)(=O)=O)C2)CCC(O)CC12CC2 C1(CN(C(C2CC(CC)C2)=O)C)CCCN1C(=O)C(C)=C1CCCC1 N1(C(=O)NC2CCCC3CCCCC23)CC2(CCC2)CCC1C(=O)O C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(O)(CNC(CC=C=C)=O)CC1 c1(C(=O)NC23CN(C(C(COC)(C)OC)=O)C(CC2)C3)cc(F)c2[nH]nnc2c1 C(=O)(CCCCCF)NC1(C2N(C(C(COC)COC)=O)CCCC2)CC1 c1(C(CC)C)ccccc1C(=O)Nc1cccc(N)n1.C1(=O)COCCN1C c1(C(=O)NCCC(=O)N(CCN(C)C(=O)C2CC2)C)ccc2nc(O)[nH]c2n1 c1(OCC)cccc(C(F)(F)C(=O)NC(CNC(=O)C=C(C)C)C2CCC2)c1 N1(CC(=O)N(c2ccccc2CC)CC)CCC(=O)N(CC)C1=O Cc1cc(C(N2CC(C(=O)NCCn3nccc3C)C2)=O)ccc1O c1(C(N(C(C)CCNC(c2ccns2)=O)C)=O)c[nH]c2cc(C(N)=O)ccc12 N1(C(C(C)N(C(C2(CC)CCCC2)=O)C)=O)CC(F)(C2CC2)C1 c1(OCCC)ccc(-c2cn(C(C)CNC(=O)CC3(O)CCOCC3)nn2)cc1 N1(C(CNC(C)=O)=O)CCC(C)(C)C1.C1(=O)CCN(C(=O)C(F)F)CCN1 C(CCC(=O)NC(C(=O)N(C)CCOCCO)C1CC1)OCC c1(-c2cn(CCN(C(CC(=O)OCC)=O)C)nn2)cccc(S(C)(=O)=O)c1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(CNC(CCCCOC)=O)C(C)(C)C1 N1(C(C2C(=C)C2)=O)CC(C(=O)NC2CNC(=O)C23CC3)CC(C)(C)C1 c1(CC(C(=O)NCC(C(C)(C)C)NC(CCC(=C)Cl)=O)C)ccc(C#N)cc1 CC1(C)CN(C(C2CC23CCCC3)=O)C(CNC(c2ncccc2CO)=O)CO1 c1(C(C(=O)OCC)NC(c2ccc(NS(C)(=O)=O)cc2)=O)ccc(Cl)c(F)c1 Cc1nc2ccc(Br)cc2cc1C(N1CCc2scc(Br)c2C1)=O c1(C(N(CC(=O)NC(c2ccccc2)CC)C)=O)ccc(C)cn1 N1(C(C2(CC=C)CCCC2)=O)CCN(C)C(CNC(C2CC2CCOC)=O)C1 c1(-c2cccc(NC(Cc3cc(C)no3)=O)n2)cc(N2CCCCC2)ccc1F c1(C(=O)NCC=CCC(=O)N(CC#C)CCF)snnc1CC C(C(C(=O)NC1CC(C)(NC(=O)Cn2cc(C(F)F)cn2)C1)NC(C)=O)OC C1(C(=O)NCCOCCOCCNC(c2cn(C)nc2)=O)CCS(=O)(=O)N1.C1CC1 c1(OC)c(Cl)ccc(C(N2CC3CN(S(=O)(=O)c4cccs4)C3C2)=O)c1F C1(CNC(C2(C)C=CCC2)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CCC12CCC2 c1(SC)ccccc1.C12(CC(NCC(=O)OC)C1)C(=O)NC2.c1(O)cnn(C)c1 C12(C(=O)NCC(=O)NCC(C)C)CC1CCN2C(=O)CC=C(Cl)Cl C(C)(CCCCC(=O)N(CC(=O)N)CC)NC(CN(CC=C)C)=O.c1(CO)ccco1 C1(CCN(C(CC)C)C)CSC(C)(C)C(=O)N1C(=O)CN1CCCC1.C(=O)O C1(CNC(=O)COCC2CC2)CC12CCN(C(c1ccsc1Br)=O)CC2 c1(C(N2CC(OC)C(NC(=O)C(F)n3cccn3)C2)=O)cc(F)c(C#N)c(F)c1 N1(C(COCC)=O)CCCC(C)(C)C1C(=O)NC1CN(C(N)=O)C1 CC(CN=c1ccc([N+](=O)[O-])c[nH]1)NC(C1CC2(CC2)C1)=O c1(C(=O)NCC2N(C(C(COC)COC)=O)CC2)ccnc(S(N)(=O)=O)c1 N1(C(C2(OC)CCC(C)C2)=O)CCCC(CNC(=O)C(C)(C)N2CCCC2)CC1 C1(NC(CC2(C)CCN2C(=O)CCc2nncs2)=O)COC2(CCC2)C1 c1(N2CC(NC(C3CC4(CCCC4)CO3)=O)(CO)C2)nc2cc(F)cc(F)c2o1 C1(CC(N2CC(n3cc(C(CC)(C)O)nn3)C2)=O)(COC)CCCCC1 C(C)(C)(CC(=O)NC1(CCOC)CCN(C(=O)C(Cc2cnc[nH]2)OC)C1)OC N1(C(c2c(C)cccc2C)C(=O)Nc2ccc(Cl)cc2F)CCCC2CCCC12 CC1=C(C)CC(c2nc(Cc3cc(F)ccc3F)nn2C2CCSCC2)CC1 c1(-c2ccc(C)o2)cccc2[nH]c(C(=O)Nc3cccc(Cl)c3)cc12 C1(C)(C(N(CCCCCC)C)=O)CCN(c2ccnc(NC)n2)C1 CCC(CC)CCC(=O)N1CCCC(C(C)NC(=O)CSC(F)(F)F)C1 c1(OC)cc(O)ncc1C(=O)N(CCCCN(C(=O)C(C)SC)C)C N1(C(Cc2c(C)non2)=O)CCN(C(c2nc(C(F)(F)F)ccc2F)=O)CC1C C(=O)(CCCc1ccccn1)NCC(C)N(C)C(C1CCC1C)=O CCC(C)C(CC)(c1nnnn1C(C)C)NC(CCCCOC)C(C)C C1(C(=O)NCC2COCCN2C(C23CCCC2C3(F)F)=O)CN2CCCN1CC2 CC(C)CCC(O)C(=O)NC(C)CCCC(N1CCCNC(=O)CC1)=O C1(NC(=O)CC2CCC(=O)N2)CCN(C(=O)CC2(N3CCCC3)CC2)CC1O N1(C(C(C(C=C)C)C)=O)CC2CCC1C(CNC(c1c(C)coc1C)=O)C2 N1(C(COC2(C)CCC2)=O)CC(C)(C(=O)NCC2(C)CC(O)C2)CC1(C)C CCS(=O)CC(=O)NC(c1ccccc1CO)CNC(=O)C(C)OC(C)(C)C CC(C)CCC(O)C(=O)N(C)CC1CCN(C(=O)Cn2cnc(C#N)n2)C1 N1(CC(=O)N(CC(C)NC(C(C)NC(COC)=O)=O)C)CCC(F)(F)C1 n1(CC)c(C)cc(C(=O)Nc2nc(Cc3cccc(OC)n3)cs2)c1C FC1(F)CC1C1CCCN(c2nccc(=NCC3CC=CCCC3)[nH]2)C1 C1(CNC(c2cccn3ccnc23)=O)CCN(Cc2ccncc2)CC1(F)F C1(SCC(=O)N(C)Cc2cn[nH]c2)CCCCC1=O C(C)(C)(C(C)CC(=O)NC1CC(n2cncn2)C1)NC(Cn1c(C)nc(C)n1)=O N1(CCN2C(CC)CCC2)CCN(C(=O)Cc2ccn(CC)n2)CC1 C1(CC)CC12CCN(S(=O)(=O)CCCN)CC2 c1(C(=O)NCC2(CC)CCN(C)C2=O)ccc2nn(C)cc2c1 N1(C(C2ON=C(C(C)(C)C)C2)=O)CCC2(CCC2NC(c2cc(O)cs2)=O)CC1 C1(CNC(c2cn(CCC3CC3)nn2)=O)CCN(C(C23CSCC2C3)=O)C1 c1(NC(C2(OC)CCSC2)=O)ccc(NC(=O)C(C)CC(C)C)cc1C C1(CC)CN(C(C2CCCCC23CC3)=O)CCN1C(c1ccc(CC)c(N)c1)=O C12(C(=O)NC3(CC=C)CN(C(C4CCCN4CCC)=O)C3)CC1COC2(C)C C1(NC(c2n(CC)ccc2)=O)CCC2(CC1)CC2NC(C1C2C3CCC(C3)C12)=O C1(N(C(N2C(C)(COC)CC2)=O)C)CCS(=O)(=O)C1 c1(CN2CC(C(=O)Nc3cnnc(Cl)c3Br)OCC2)ccc([N+](=O)[O-])cc1 c1(CC(=O)NCC#CCNC(C2C(CC)C2)=O)cc(S(N)(=O)=O)cn1C C1(NC(C2C(C)(CC)C2)=O)CCSC12CN(C(=O)C=Cc1cccc(CO)c1)C2 c1(C(N2C(C(=O)NC(CCN(C)C)(C)C)CC2)=O)cncc(C#N)c1 Cc1ccc(C(C(=O)NCCC2CCCN2C(=O)CCCF)C2CC2)cc1 Cn1cnc2ccc(CCNC(=O)C(N3CCOCC3CC(F)(F)F)=O)cc12 C1(C(N2CCN(C(C(C(=C)Cl)(C)C)=O)CC(O)C2)=O)Cc2nn[nH]c2C(C)C1 Cc1cccc2c(C(N3CCOC(CC(=O)NC(CO)C(C)C)C3)=O)n[nH]c12 CCC(C)C(C(=O)NC1CCCC1C(=O)NCc1ccc(C(=O)OC)o1)OC c1(C(=O)NC(C2(O)CN(C(c3c(COC)nn[nH]3)=O)C2)C)cnc2cccnn12 C1(C(=O)OC(C)(C)C)CCCCC1N=c1[nH]c2cc(Br)ccc2o1 C1(C(=O)Nc2ncc(C(C)=O)cc2C)CCc2nnc(O)n2C1 N1CC2CCN(C(=O)Cc3ccc(Cl)s3)C2C1.O=C1CCCN1CCO CCC(CC)(CCOC)C(=O)NC1CC(NC(=O)CCc2cc(C)on2)C(O)C1 N(C(=NCCc1ccnc(Cl)c1)NC(C1CC1)C1CC1)C1C(F)C1 C1(C(=O)NCC2CN(C(C3C(C)(Br)C3)=O)C2)Cc2cc(F)ccc2C(=O)O1 c1(COC)cc(C(=O)NC2CCCC2NC(=O)C=Cc2cc[nH]c2)n(C)c1 C1(OC)C(NC(=O)NNC(c2cc(Cl)ccc2C)=O)COC1(C)C c1(C(=O)NCC2(NC(C(C)CF)=O)CC2)noc2c1COCC2 C1(n2cccn2)(CNC(C(CSC)O)=O)CCN(C(C2CCC2C(F)F)=O)CC1 N1(C(=O)OC(C)(C)C)CCOC(C)(CNC(=O)CCS(C)(=O)=O)C1 c1(C(N(CC(C)NC(c2c(CC)cccc2F)=O)C)=O)ccc2c(c1)C(C)CN2 n1(C(C)C)cc([N+](=O)[O-])c(=NCC2CCCN(C(C3CC=CCC3)=O)C2)[nH]1 C(C(CC(C)C)C(=O)N(C)C(C1CC1)C1CC1)NC(CCCCOCCOC)=O N1(C(C(C)(C)N2CCCCC2)=O)CCC(CO)(NC(C2CC2C(N)=O)=O)CC1 C1(NC(C2C(C)OC(C)C2)=O)(CO)CCCN(C(c2cn(CCO)nn2)=O)C1 N1(C(COc2c(OC)cccc2)=O)CC(NC(=O)C=Cc2cnc[nH]2)C(C)(C)C1 N1(C(c2ccc(C)cc2)=O)CC(C(=O)NC(C(N)=O)C2CC2)OC(C)C1 c1(C(=O)NC(CNC(C(F)=CC)=O)CCOC)sc2cccc(Cl)c2c1Cl c1(C(=O)OC)cccc2oc(=NCCCCNC(=O)C(C(C)C)NC=O)[nH]c12 N1(C(CC(=O)OCC)=O)CCC2(CCC(C(=O)NCc3ccnc(Cl)c3)C2)CC1 C12(C(=O)NCC(C=C)(C)C)CC(CO)(CN1C(=O)CCNC(=O)OC)C2 C1(CNC(C(C)OCCCC)=O)CC(O)CN1C(c1nc(C)nn1C)=O C(CCCC(=O)NCCCC(C)NC(=O)CC(c1ccccc1C(F)(F)F)C)OC C1(CNC(C2(CC)CC2)=O)CC12CCN(C(c1cc(C(C)C)ccc1C)=O)CC2 CCC(C)(CNC(c1cc(OC)no1)=O)C(=O)N1CC(OC)CC(C)C1 N1(C(c2cccc(CC(C)C)c2)C(=O)NC2COC2)CC(C)CCC12CC2 c1(CC)cc(C(=O)NC2CCCC2C(=O)NCCNC(=O)NC)c(F)cc1C C12(C(=O)NCC(C3CCN(C(C45CC4C5)=O)CC3)(C)C)CCC(F)(CC1)CC2 CC1(NC(C2CCCO2)=O)CCN(C(=O)CCCCNC(N)=O)C1 C1(C(N2CCC(N(C(CC3CCC(C)CC3)=O)C)CC2)=O)CC2(C1)CC(O)C2 C=C(Cl)C(C)(C)C(=O)NCC1CCCCN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 c1(CC(=O)N(C(C)CNC(C2(O)CC2C(F)(F)F)=O)C)nc(F)ccc1Cl C1(C(N2CCCC(N(C)C(c3cnn[nH]3)=O)CC2)=O)CC(=O)C12CCCC2 c1(NC(C(C)CC2CCCO2)=O)ccc2ccn(CC(=O)N(C)C)c2c1 C1(C)(C(=O)NC(C(=O)OC)O)CCCN1C(=O)CC(c1cccs1)c1ccc[nH]1 N1(C(c2c(C)occ2)=O)CCC2CCN(C(C3CCC(N=[N+]=[N-])CC3)=O)CC2C1 N1(C(C(N2CCCC(N(C)C)C2)=O)=O)CCc2cc(Br)cc(Cl)c2C1 N1(C(C2C(CN(C)C)C2)=O)CCC(CNC(c2coc(C(C)(C)C)n2)=O)C1(C)C Cc1ccc(C(=O)NCCC2(C(=O)NCC3(O)CCOCC3)CC2)cc1O N1(C(C=Cc2ccn(C)c2)=O)CC(C)(C)CCC1CNC(c1cnco1)=O c1(CC)c(C(=O)NC2N(C(c3ccccc3)=O)CC2(C)C)cnn1C.C(=O)OC CCC(C)CCC(=O)NCc1ccc(CN(C)C(C2(F)CC=CCC2)=O)cc1 CC1CN(C(=O)C(Cl)Cl)CC1(C)C(=O)NCC1(C(C)O)CC1 CC1(C(=O)NC(CNC(C2(C(F)(F)F)CCOCC2)=O)C(C)(C)C)CC(F)(F)C1 C(C(C)C(C)C(=O)N(C)CC1CCN(C(C2CC(OC)C2)=O)CC1)OC N(C1CCCc2ccc(Br)cc21)C(C1C2(CN(C(c3ncsc3Br)=O)C2)C1)=O c1(CC(=O)NC2(C3CN(C(C4C(C)(C)C4)=O)C3)CC2)cccc2sccc12 N1(C(CC(CC)C2CCC2)=O)CCN(C(c2cc(C(C)C)on2)=O)C(CCO)C1 c1(OC)cccc(CNC(=O)NC2CC(C)(C)O2)n1 C1(NC(c2cnc(OC)nc2)=O)CC2CC(NC(C3COC3)=O)CC2C1 C1(C(=O)NC(CC)CO)CCCCC1NC(=O)COCCCOC C1(NC(CCc2nc(C)c(C)[nH]2)=O)CC2CCC(C1)N2c1ncnc(=N)[nH]1 N1(C(c2scc(C)c2C)C(=O)NCCCSCC)CCC(O)C(C)(C)C1 c1(CNC(=O)NCC2N(C(=O)OC(C)(C)C)CCC2)ccc(Cl)cn1 N1(C(c2c(CC)csc2)=O)CC2(C(=O)NCC(c3nccs3)C)CCC1CC2 N1(C(C=CC(=O)OC(C)(C)C)=O)CC2(CCC(CNC(=O)CC3CC3)O2)C1 Cc1ncc(C(N2CC(Cn3cc(C4(C)CC4)nn3)C2)=O)c(C)n1 N1(CC)CCOC(C(=O)NC(Cc2cnn(C)c2)C(=O)NCCO)C1.C1CCO1 N1(C(c2occ(OC)c(=O)c2)=O)CCCC2(CCC2NC(=O)CC2CC2)C1 C(=O)(C(CC(=O)N(C(C)CNC(C12CC(C)(CO1)C2)=O)C)C(C)=O)OCC N1(C(c2c(CC(C)C)ncs2)=O)CCC(C)C(NC(=O)CCN(C(=O)NC)C2CC2)C1 C(=O)(C#CC1CCC1)NC1CC(C(C)NC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 C(=O)(C(Cc1ccsc1)NC(=O)C(C)N)OC CCCCC(CNC(c1snc(Cl)c1Cl)=O)Nc1cnc(C(=O)NC)cn1 CC(Cc1ccccn1)C(=O)NCCC(C)NC(c1cc(Cl)cs1)=O C(=O)(C(C)(F)C(C)(C)F)NCC(C(C)(C)C)NC(c1ccc(C#N)cn1)=O c1(NC(N2CC(CC(=O)OCC=C(C)C)C2)=O)cnn(CCl)c1.C(C)(C)(C)S c1(N(C(CC(C)(C)C#N)C(=O)NC2CC2)C)ccc(C#C[Si](C)(C)C)cc1 CN1CC(C)(C(=O)NCC2CCCN2C(c2cc(C(F)(F)F)ncn2)=O)CC1=O C(=O)(CC(C)(O)COC)N(CCCNC(=O)Cn1nnc(-c2ccsc2)n1)CC C#Cc1ccc(C(=O)NCCC(C)(C)NC(c2nc(O)sc2C)=O)c(F)c1 Cc1c(C(N2CCCC(C(=O)NCCS(C)(=O)=O)CC2)=O)ccnc1Cl CCC(CC(=O)N1CC(CNC(c2ccc(-c3nccs3)cc2)=O)C(O)C1)OC c1(C(=O)NCC(O)CCNC(C2C3COCC23)=O)nc2c(s1)COCC2 CC1CC(C)N(C(=O)CSc2ccccc2)CCN1C(c1cc(O)nc(Cl)c1)=O C1(CC=C)(NC(c2cnc(C3CC3)nc2)=O)CCN(C(=O)C(C)n2cncn2)C1 c1(C(=O)NC2CCN(C(COC)=O)C2)cnc2c(c1)CCC(=O)N2 N1(C(CC2(C)CC2)=O)CSCC1C(=O)NCC1(F)CC(O)C1 N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCCN2C(C)=O)=O)C1 C1(C(N(C2CC(SC)C2)C)=O)CCC(O)CN1C(=O)Cc1cccc(F)c1 c1(OC)cc2ccccc2cc1C(N1CC(N(C(=O)CC2CCC(=O)N2)C)C1)=O N1(C(C(C)(F)F)=O)CCC2(CC1)CC2C(N1CCCCC(F)(F)C1)=O c1(NC(C(C2CCN(C(c3ccncn3)=O)CC2)C)=O)nc(Cl)ccc1I N1(C(CC(=C)C)=O)CCCCCC(NC(c2cc(C)cc(C)c2C)=O)C1 Cc1cncc(C(=O)NCC(N2CC(NC(C3CC(C(C)(C)C)C3)=O)C2)=O)c1C CC1(C)CC(NC(=O)C=Cc2cnc[nH]2)CN1C(c1cccc(N)c1)=O c1(OC)cc(C(=O)NC2CN(C(=O)CCC3CC3(F)F)CC2OC)ccc1Cl C12(CCNC(CC3C(=O)NC(=O)N3)=O)CCC1CN(C(=O)C(=O)NC1CC1)C2 N1(C(CC(C)n2cccn2)=O)CC(C2(NC(=O)CN3CCCCC3)CC2)C1 n1(CC(N2CC3C(CNC(c4cc5sccc5[nH]4)=O)(C3)C2)=O)ccc(O)nc1=O Cc1nccn2c(-c3nc(C(C)O)nn3-c3ccc(Br)nc3)cnc12 N1(C(C2N(C(C(CC)n3cncn3)=O)C3(CC2)CC3)=O)CC(O)C(O)C12CCC2 C1(C)(C(=O)NCc2occ(C(N(C)Cc3ccoc3)=O)c2)CCC2CC2C1 Cc1cc(C)cc(C=CC(=O)NCCOCCNC(c2ccccn2)=O)c1 c1(C(N2CCOC(CN=c3[nH]nco3)C2)=O)ccn2ccccc12 C1(C(=O)NCCN(CCOC)C(c2csc(CO)n2)=O)CCC(=O)NC1 c1(NC(C2(OC(CNC(c3ccc[nH]3)=O)=O)CCC2)=O)cc(F)cc(Br)c1O N1(C(C(C(C)NC(c2cc(C(N)=O)co2)=O)C)=O)CC(O)(C2CCC2)C1 c1(OC)ccc2c(c1Br)C(NCCCc1ncccn1)CC2 C(=O)(CC(=O)N1C(C(=O)NC(c2ccncc2)(C)C)CC1C)NCC N1(C(c2ncn(C)n2)=O)CCC2(CCCC2NC(=O)CCn2ccccc2=O)C1 N1(C(c2c(C(C)C)n[nH]c2)=O)CCC2(CCN(C(C3CCC(C)O3)=O)CC2)C1 c1(CC(N2CC(N(C(COCCOCC)=O)C)C2)=O)c[nH]nc1O c1(NC(C2(C)CN(C(C(C)OC)=O)C2)=O)cnc(Cl)nc1C c1(C(N2CCCC(C)(NC(CNC(=O)NC)=O)C2)=O)cccc2nc(C)nn12 C1(C2C(C)C2)CCC(NC(=O)CCn2cccn2)C1.C1CC(Cl)=CC(=O)N1CC C=Cn1nccc1C(N1CC(NC(c2scc(OC)c2OC)=O)CC1CO)=O C1(NC(c2c(C)noc2)=O)CC(F)CN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C1 CC(CC(=O)NC1CCC(NC(=O)CNC=O)C1)C1CCCC1 N1(C(CCCC)=O)CCSCC1CCNC(c1ncoc1-c1ccc(C)cc1)=O C1(CC(=O)NCC(CC)(C)NC(c2cscc2F)=O)CC=CCN1C CC1CCCC1(C)C(N1CCN(C2CN(C(=O)Cc3nc[nH]n3)C2)CC1)=O C1(C(N(C)CCn2cnnc2)=O)CCCCC1NC(=O)C=C(C)C(C)C C1(CNC(C(=O)NC(C)C)=O)CC2CC(C1)N(C(c1noc3c1COCC3)=O)C2 c1(C(N(CCN(C(C2SCCCS2)=O)CC)CC)=O)cnn2c1N(C)CC2 C(=O)(C(C)N(C(C1CN(C2COC2)C1)=O)C1CC1)N(CC)CC N1(CC2C(c3n4c(nn3)C(=O)OCC4)C2)CCC2(CC1)CC(n1cncn1)CCO2 C1(C2CCN(C(C(c3cc(OC)c(=O)n(C)c3)=O)=O)CC2)NC(=O)N2CCNCC2C1 C=CCCCCCC(=O)NCCCCC1(NC(C2(C)CCC(F)(F)C2)=O)CC1 n1(CC(=O)NCCc2ccc(C)o2)cc(Nc2oc(C)nc2C)c2ccccc12 N1(C(C2C(COC)C2)=O)CC2CC1CN(C(c1cc3occc3n1C)=O)C2 C1(NC(CC2(C(=C)F)CCC2)=O)CC2(CCN(C(c3cccc(N)c3)=O)C2)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)N(C)CCN.C12(C=O)CCC(CC1)C2=O C1(NC(c2c(C(C)C)c[nH]n2)=O)CN(C(c2cc(C(F)F)n(C)n2)=O)C2CC12 CC1(C)CCOC(C(=O)NC(C2CCCCC2)CNC(c2ccc(Cl)cc2)=O)C1 c1(OC)nc(C)ncc1C(=O)NC1CN(C(c2ccc(C(C)(C)C)[nH]2)=O)CC1C CC1Cc2cccc(C(=O)NCC(O)CNC(C3Cc4nccnc4C3)=O)c2O1 Cc1cn2nc(N3CC=C(CCNC(C4(F)CCS(=O)(=O)C4)=O)CC3)sc2n1 C1(NC(c2c(OC)ccs2)=O)CN(C(c2cc(O)nc(Cl)c2)=O)C2(CCOC2)C1 CCCC(CC)CCC(=O)NC1CCN(C(=O)CNC(=O)CC(C)(C)C)C1C CN1CC(NC(=O)CCCCCNC(=O)CC(=O)NC2CC2)CC1(C)C C1(C(=O)NCC(C)O)CC2(CCN(C(=O)Nc3ccc(C(N)=O)cc3)C2)C1 c1(C(=O)NC(C(CC)C)C(=O)OC(C)(C)C)nccc2n[nH]cc12 C(c1cn(C)cn1)=CC(=O)NC(CCN(C)C(c1nccn1C)=O)(C)C N1(C(C(C(C)C)C(C)C)=O)CCC(C2(NC(=O)CCc3ccoc3)CCC2)CC1 C=C(Cl)CC(C(=O)NC)NC(=O)C(C)NC(=O)CCC(C)(C)F NS(=O)(=O)c1cc(C(N2CCCC3(C2)CN(C(c2cnsn2)=O)C3)=O)c(Cl)o1 N1(C(C(C)CC(N)=O)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)C(F)(F)F)C1 CC(C(=O)NC1CC2(C1)CC(NC(C1OCCN(C)C1=O)=O)C2)C(C)(C)C c1(C(N(CC(C)(C)NC(Cc2ccc(C)c(Cl)c2)=O)C)=O)cc(Cl)cc(F)c1F Cc1cc(OCC(N2CCCC(NC(c3n[nH]c(C)c3C)=O)C2)=O)cc(C)c1Cl C(CC(=O)NCC(C)N(C(=O)Cc1sc(C(C)OC)nc1C)C)(C(C)C)OCC C1(NC(C2(c3ccc(OC)cc3)CC2)=O)CN(C(=O)CC2CSC2)CCC1CO N1(C(c2ccc(OC)cc2F)=O)CCC2(CC1)CN(C(=O)CC1CCSCC1)C2 C1(NC(c2cc(CCC)[nH]n2)=O)CC(O)CN(C(C2(CC)COC2)=O)C1 c1(CC)csc(-c2ccc(CC(=O)Nc3c[nH]nc3CC3CCOC3)s2)n1 C(=O)(CCCCCCC(=O)NC(Cc1ccccc1[N+](=O)[O-])CO)OC CCC(C)C(O)C(=O)NC1CN(C(=O)Cc2ccc(C#N)nc2)CC1C c1(NC(C2N(C(C3(C(C)C)COC3)=O)CSC2)=O)ccc(O)c(=O)cc1 N(C1CCCc2ncccc21)C(=O)NCC1CCCC1 C1(O)(CNC(Cc2scc(C)c2)=O)CCN(C(C2CC(CN(C)C)C2)=O)C1 c1(CNC(=O)NCC(CCCC)CCC)ccc2c(c1)OC1(CCC1)O2 C1(C(N2CCC(N(C(=O)CO)C)C2)=O)CCc2c(ncn2C)C1 S(=O)(=O)(c1cccs1)NC1CCN(C(c2ccccc2OC(F)F)=O)CC1F C1(N2CCCC(C)(O)CC2)CC2(CCN(C(=O)C(=O)NCCC3CC3)CC2)C1 N(C1CC(C)n2ccnc21)C(=O)NC1CC(c2ccccc2)(C(=O)OCC)C1 Cc1cc(C(=O)N(C)CCNC(C2CC2(C)Br)=O)cnc1C(F)F c1(NC(CCCSc2nnc(C(=O)OC)s2)=O)ccc(CF)cc1 CS(=O)(=O)C1CN(C(=O)C=Cc2ccncn2)CC1C(=O)NCC1C2CC3C(C2)C13 C(=O)(CCCC(C)(F)F)N(C)CC1(O)CN(C(C2CC(C)OC(C)C2)=O)C1 N1(C(C(CC=C)CC)=O)CCOCC(C)(CNC(=O)CCc2cc(Cl)cs2)C1 N1(C(c2c(C)nc(O)s2)=O)CC2CC(NC(c3cc(F)ccc3Cl)=O)CC1C2 c1(C(=O)NCC2CCN(C(c3ccco3)=O)CC2)cccc2c1CCO2 CCC(C)(C)CCCC(=O)N(C(C)C(=O)NCCOC)CC.C1CCO1 c1(CC(=O)NC(C)(CNC(C2(O)CC2)=O)C2CC2)ccc(Br)s1 C(CCC(C)C(=O)NC1CCC(CNC(c2occc2C(C)C)=O)CC1)OC Cc1cc(C)c(CC(=O)NC2CCN(C(c3cn(C)c(O)n3)=O)CC2)s1 Cc1cncc(C(=O)NC2CCN(C(c3ccc(N(C)C)cn3)=O)C2)n1 C(C)(CN=c1[nH]c(C)cc(=NCCCC(C)(F)F)[nH]1)Oc1c(OC)cc(OC)cc1 N1(C(c2cccc(C)n2)=O)CCC2(CCCCN(C(=O)Cc3scnc3C)C2)C1 C1(COC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CC1(C)CC1 N1(C(c2cscn2)=O)CCN(C(=O)Cc2ccc(O)c(F)c2)C2CC12 c1(C(N(CCCNC(Cc2scc(C)n2)=O)C(C)C)=O)ccc(O)cn1 C1(CNC(COC)=O)CC(F)CN1C(=O)C(C)CC1CC1 c1(C(=O)N)ncc(P(C)(C)=O)cn1.N1(CC(=O)NCC(C)CC)CCCOC1=O c1(C(=O)NCC(CNC(C2(CC=C)CC2)=O)(C)O)cc(OC)ncc1F N1(C(C2OCC(C)(C)C2)=O)CC2(CCNC(c3ccc[n+]([O-])c3)=O)CCC1CC2 C1(NC(C2(CC#C)CCCO2)=O)CCN(CC(=O)NC2CC2)CC1 N1(C(C=CCCC)=O)CCOC(CCNC(=O)Cc2ccc(C(=O)NC)s2)C1 C(C)(CC)(C(=O)OC)NC(CCC1(C)CN(C(C=C(CC)C)=O)C1)=O c1(C(N2CCN(C(c3nc(C)sc3C)=O)CC2)=O)cc2c(nn1)CCC2 CC1(C)CCOC1CCC(N1CCC(C(=O)NC(CO)C2CC2)C1)=O N1(C(COCC#C)=O)CC2(CC(NC(=O)C=C(C)c3ccccc3C)CO2)C1 c1(C2C(C(=O)NCC(=C)CCNC(=O)CC3CC4CC4C3)C2)ccc(F)cc1 c1(C(=O)NCC2CCN(C(COCCCC)=O)CC2)cccc(C#CC2CC2)c1 Cc1cn2c(C(N3CC=CC3CNC(=O)COCC(C)C)=O)cnc2s1 C1(NC(C(CC)C)=O)CN(C(c2ncccc2O)=O)CC2(CC2)C1 C(CC(=O)NC(=O)CSCC1CCCO1)SCCC1(OC)CC1.C(C)N c1(CN(C)C)ncc2c(n1)CCN(N1CCN(C(=O)OC(C)(C)C)CC1)C2 Cc1cc(F)ccc1S(=O)(=O)N1CCNC(C(=O)NCc2cocn2)C1 CCCC(C(=O)Nc1cnsc1)NC(=O)C(Cl)Cl C1(NC(CC2CCC(C)C2)=O)CCC2(CC1)CN(C(C1CCN1C)=O)C2 S(=O)(=O)(c1cn(C)c(=O)n(C)c1=O)NCCc1ccc(NS(C)(=O)=O)o1 C1(NC(CC(c2ccc(C)cc2)C)=O)CN(C(C2(C)CCC2)=O)CCC12CCC2 C(c1c(Cl)nc2sccn12)=CC(N1CCC2C(C1)CN2C(=O)CSC1CC1)=O C(CC(C(=O)NC(C1CCC1)C)NC(=O)Cc1cnn(C)c1C)SC C(=O)(C(C)(C)CC(=O)N1CCC2(CC1)CC2C(=O)OC)NCCC(=O)OC C1(CNC(C(C=C)OC)=O)CCN(C(c2ccccc2)=O)C1(C)C c1(CCC(=O)NCC(CCOC)NC(c2nc(C)nn2C)=O)ccccc1C C1(CC)CCCN(C(=O)COC2CCN(C(c3sccc3C)=O)C2)C1 Cc1nn(C)c(C(=O)NCC2(NC(=O)C(C)(C)n3cnnn3)CC2)c1[N+](=O)[O-] C1(NC(CNC(C2C(C)C2)=O)=O)CC2CN(C(=O)C(F)(F)C3CC3)CC2C1 C1(CC)CCN(C(=O)C(C)(C2CCC2)NC(=O)C(O)C(C)SC)CC1 N1(C(C(CC)COC)=O)CC2(CC2)CC1CNC(=O)Cc1ccccc1C(N)=O N1(C(CCC=C)=O)CC2(C1)C(NC(=O)Cc1nc(C)sc1C)CCS2(=O)=O C(C)(C(=O)OC(C)(C)C)(C(=O)N1CCCC(NC(=O)C(F)OC(F)(F)F)C1)OC C1(NC(c2cc(COC)c(F)cc2)=O)CC2CN(c3ncc(OC)cn3)CC2C1 Cc1cc(C)c(C(=O)NC2CCN(C(=O)CNC(=O)C3CC3)CC2F)c(O)c1 C1(NC(C2(CC)CCCC2)=O)CC2CCCC(C1)N2C(=O)Cc1cnoc1 N1(C(CC(C)(F)F)=O)CCC(CCNC(=O)CCCCC#N)C(F)(F)C1 c1(C(=O)NC(C2(O)CN(C(C3CCCS3)=O)C2)C)cc2c([nH]1)CCC2 N(C1CCCc2c1cnn2C)C(=O)NC(C(=O)NCCC)CC CC1CN(C(C2CCC=CCC2)=O)CC1CC(=O)NC1CCC1(C)C C#Cc1cccc(C(N2CCN(C)C(CNC(C3CS(=O)(=O)C3)=O)C2)=O)c1 C(C(C(=O)N(C(C)CN(C)C)C)NC(=O)CC1CC=CCC1)OC C(CC(O)C(=O)NCC1COCCN1C(=O)CCc1ncc(Br)cn1)SC C=CC(F)(F)C(=O)NC1CC(C)N(C(c2cccnc2NC)=O)C1 c1(CN2CC3CN(C(c4c(C(C)(C)C)[nH]cn4)=O)CC32)n[nH]c2ccc(Cl)cc12 c1(C(N2CC(CNC(C3(CC#C)CCOCC3)=O)C2)=O)cc(C)nc(Cl)c1N CC1(C)C2CCC(C2)C1C(=O)NCCC1CCCN1C(=O)CCNC(=O)CO CN1CCC(C)(C(N2CCCC(c3cn(CC4COC(=O)C4)nn3)C2)=O)CC1 C1(C(=O)NCC2C(CNC(C(C)N=[N+]=[N-])=O)C2(F)F)CNC(=O)CC1C c1(CNC(C(C=CC)O)=O)ccc2c(c1)CN(C(c1ccc(F)c(F)c1C)=O)C2 CCCC(C)(O)CC(=O)NC(CC(=O)N1CC2C(C1)C2(F)F)C(C)OC C(=O)(C(COC)CC(C)C)N1CCC(O)(CCNC(C2(C=C)CCC2)=O)CC1 N1(C(c2cccc(C)c2F)C(=O)N(C(CC)(C)C)CC)CC2CCC(C1)C2(F)F c12cc([nH]n1)C(=O)N(CC=C)CCC(=O)N2.C(COC)(C(C)C)SC C(=O)(C(C)C1=CCCC1)NC1CCN(C(c2cc(C)oc2C)=O)CC1O N1(C(Cc2cc(C)on2)=O)CCC2(NC(=O)CSC3CC3)CCCCC12 C(CCN=c1nc2ncn(C)c2c(NC2CN(C)C3(CCC3)C2)[nH]1)n1ncc(C)c1 CCC(CC(F)F)C(=O)N1CC(O)(CNC(c2ccc(C)c(O)c2)=O)C1 N1(C(C(N2CCOCC2)C)=O)CCCC1(C)CNC(c1ccsc1)=O C1(C(=O)NCc2n(CCC)ccn2)CCC2CCC1N2C(=O)CC1CCCO1 c1(NC(C2(F)CCN(c3nc(C4CC4)ncc3Br)C2)=O)ccnc(Cl)c1Cl C12C=CCN1C(=O)CNC2=O.c1(C2(CNC(c3ccccn3)=O)CC2)ccccc1 C1(=CC(N2C3CN(C(CCCOC)=O)CC2CC3)=O)CCOc2ccccc21 c1(CN(C)CC2CNC(C)(C)C2)cccc(OCC(F)(F)F)n1 C1(C(=O)NCCC2CCSC2)CCCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(C(=O)NCCN(C(c2c(C)[nH][nH]c2=N)=O)C)cc2cccc(F)c2o1 CC1(C)OCc2cc(C(=O)OCc3cnn(-c4ccccc4)c3N)ccc21 c1(C2(C(=O)NC3(CNC(c4c(C)nc[nH]4)=O)CCOC3)CCC2)ccccc1Cl c1(C(=O)NCC23CC2CN(C(c2cc[nH]c2)=O)C3)cccc(Cl)c1Cl O=C(C1CCSc2ccccc21)NC1C2CC1N(C(C1CC3CCC1C3)=O)C2 C(=O)(C(CO)C(F)(F)F)NC1CCCCN(C(CCC(C)(F)F)=O)C1 C(=O)(CC(C)CC(=O)N1CC2CCC1CN2C(C1(NC(C)=O)CC1)=O)OC N1(C(=O)Cn2cc(C3CCCC3)nn2)C2CCC1CC(CC1OCC(C)C1)C2 c1(CC)cnn2ccc(C(=O)NCCC(C)NC(c3cc(C)[nH]n3)=O)nc12 C12(C(=O)NCC3N(C(c4n(CC)ncn4)=O)CCOC3)CC1COC21CCC1 c1(CNC2CCN(C3CCC(C)CC3)CC2)ccnc2ncccc12 C1(CC)C(NC(c2coc(-c3cccc(F)c3)n2)=O)CCN1C(=O)CC(O)CC Cc1ncccc1-c1cn(CCNC23CC(C(C)(C)C)(C2)C3)nn1 c1(CC(=O)N(C2CCCN(C(=O)Cc3cccs3)C2)CC)cc(F)c(F)cc1F C1(CNC(CC=C(C)C)=O)OCC2CCC1C2.C12C(C1(C)C)NC2=O CCC(C(=O)NCC1CC(F)(CNC(=O)Cn2nnc(=O)[nH]2)C1)C(F)(F)F c1(C(N2C(CNC(C3CN(c4nncs4)C3)=O)CCCC2)=O)c[nH]nc1[N+](=O)[O-] c1(OC)cccc(C(C(=O)NC2(C)CC(C)(C)C2)N(C)Cc2ccc(F)cc2)c1 c1(CC(=O)NC(C)CN(C)C(C2(C#N)CCC2)=O)nn(C)c2ccccc12 C12(C(=O)NC3C(NC(c4nc(COC)sc4)=O)CCCC3)CC3CC(CC1C3)C2 c1(C(=O)NC2C(C)N(C(=O)CCC(=O)N(C)C)CC2)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2n(C)ccn2)=O)CCN(C(C2CCCCNC2=O)=O)C1(C)C C1(NC(=O)COc2cn[nH]c2)CC(F)(NC(C2CN(c3ccccn3)C2)=O)C1 C=CCC(CC)C(=O)N1CC2CC2(CNC(=O)Cc2cnccc2Cl)C1 c1(CC(=O)NCC(C2CCOC2)NC(C23CCCN2CCC3)=O)cc(F)ccc1Cl c1(CC(=O)NC(CNC(CCC(=C)Br)=O)C(C)(C)C)ccc(O)c(Cl)c1 C1(CNC(C2(CCC=C)CN(C(n3nc(C)nc3C)=O)C2)=O)CC2(CC2)C(=O)O1 C12(C(=O)NCCOCCNC(CC(CC)C3CC3)=O)CCC(CC1)C2(C)C c1(C(=O)NC(C)C(C)NC(=O)Cc2cn(C)nc2Cl)cccc2c1CNC2=O N1(C(c2c(C)con2)=O)CCC2(CCCC2NC(C2(F)CCCCC2)=O)C1 O=S(=O)(c1ccnn1C1CC1(F)F)Nc1cnn(-c2ccccc2)c1 CC(O)C(C)(C)C(=O)N(CC(O)CNC(=O)CC1CCN(C)C1)C C(=O)(C1=Cc2ccccc2C1C)N(CC)CC1CCCN1C(=O)C(F)(F)C(C)O C1(c2nnnn2CCC2(C)CC2)(N(C(CCCCCC)C)CC)CC2CCC1CC2 c1(C(=O)NC(CN(C(=O)C=NOC)CC)C)ccc(-c2ccc(Cl)cc2)cc1 C1(C(N(CCNC(C2(C)CC=CC2)=O)CC)=O)CC(O)CN1C(=O)OC(C)(C)C C(N=c1[nH]c(=NCCCN2CCC2)[nH]c2c1CSC2)c1nc(CC)sc1 N1(C(c2c(C)nco2)=O)CC(NC(C2(C)CC(C)(C)C2)=O)CC12CCOCC2 C1(NC(Cc2cc(C)sc2)=O)CC2(CCN(C(=O)C3CC3)C2)C1 c1(C(=O)NCCCC(C)NC(c2ncoc2C2CC2)=O)cnc(Cl)c(F)c1N CCC(C)CC(=O)C(=O)N1CC2CC(C(=O)NOCCC(C)O)C(C2)C1 CCCCCCCCCC(C)CC(=O)N1CC2CCC(C1)N2C(C1SCCS1)=O C1(=CCNC(C(COC)O)=O)CCN(C(C2CCCCS2)=O)CC1 C(C1c2ccsc2CCN1C(C1CCCCC1)=O)NC(CC1(C)CCC1)=O C1(C(=O)NC2CN(C(c3cnc(N(C)C)n3C)=O)C2)CC2CCCCN2C1 N1(C(=O)OC(C)(C)C)CC2CCC2(C(=O)NC(c2nn[nH]n2)C2CC2)C1 C1(CC(=O)NCC(C)=CC=O)CCOCC1.C(C(C)(C)C)NC(C)C Cc1ccc2c(c1)CCC(C(=O)NC1CCN(C(C3CCOC3)=O)C1C)O2 N1(C(c2cc(CCNC(CC=C=C)=O)on2)=O)CCC(C)(C#N)C1 c1(C(N2CC3CCN(C(c4c(C)nn(C)c4)=O)C3C2)=O)cc(F)cc([N+](=O)[O-])c1 Cc1c(C(=O)N(C)CC2CCCN(C(=O)CCn3cncn3)C2)ccc(F)c1F C1(NC(C(CC#C)C2CC2)=O)CCCN(C(=O)C(C)Cc2ccccn2)C1CC C1(NC(c2cc(C)c(C(F)F)nc2)=O)CCCN(C(c2sccc2Cl)=O)CC1F c1(CC(=O)NCC(CC)NC(c2cnc(COC)s2)=O)cc(C)cs1 CC1CCN(C(=O)CCCCCN(C)C)CCN1C(C1CCCCCS1(=O)=O)=O Cc1nn(C)c(C)c1C(N1CC(C(=O)NCC(C)(C)C(C)(C)O)C(C)C1)=O N1(C(CC(C)C2CCCCC2)=O)CC2(C1)CN(C(c1ccc([N+](=O)[O-])s1)=O)C2 CC1CN(C(=O)CCCN2CCOCC2)CC1CNC(c1cccs1)=O N1(C(c2cccc(CC(C)C)c2)=O)CCC(C)C(NC(=O)COCC(F)F)C1 N1(C(C2CC=CCN2C(c2cc(CO)on2)=O)=O)CCC(CO)C(O)C1 C(=O)(CC(O)(CC)c1ccccc1)NC(CC)CNC(c1nc([N+](=O)[O-])n[nH]1)=O Cc1ccc(F)c(CC(=O)NC(C)(CNC(C2(O)CCCCC2)=O)C2CCC2)c1 C(=O)(C1=CC2C=CC1C2)NCCCN(C(C1CC(CCC)C1)=O)C(C)C Cn1ncc(C(=O)NCC2CCCN2C(C2CCCCO2)=O)c1C(F)F C12(C(N3CC(C(C)NC(COC(CC)(C)C)=O)C3)=O)CC3CC(C1)CC(C)(C3)C2 c1(N2CCC(OCCOC)C2)nc(C)cc(=NC(C)CN2CCOCC2)[nH]1 N1(CC)CC(C(=O)N(CC(C)(C)CNC(c2csc(C)c2OC)=O)C)CC1=O C1(NC(=O)CCOC2CCC2)CC2(CCN(C(=O)CC3CCCCCO3)CC2)C1 N1(Cc2cncc(OC)c2)CC2CCC1CN2C(c1ccc(C)cc1)=O CC(C)CC(C)C(=O)N(C1CCN(C(c2coc(C3CCCC3)n2)=O)C1)C c1(CC(N2CCC(C(C)NC(c3c(CC)occ3)=O)C2)=O)cc2ccccc2o1 c1(C(N2CCC2Cc2c(-c3cn(CCC)nn3)n(C)nc2)=O)c(C)cccc1Cl c1(N2CCC(OC)C2)nc(=NCCC(COC)CC(C)C)[nH]c2c1CC(C)CC2 c12ccc3c(c1)CN(C3)C(=O)C1C(C1)C(=O)N2.c1(OCC)nc(Br)c(Br)cc1Br c1(C(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)F)c(F)cccc1F C1(NC(c2c(C(C)NC(=O)CCN3CCOC3=O)noc2)=O)CC2(CCC2)C1O C1(CC(=O)NCC(C)(C)C(N)=O)CCCN(C(=O)CCc2cn[nH]c2)CC1 c1(C(=O)NC(CNC(C(C)OCCOCC)=O)C)cc(C)nc(Cl)c1N c1(C(=O)NCCNC(=O)Cc2ccc(F)cc2C(F)(F)F)cnc2n1CCCC2 CC(C)C(CO)C(=O)NCC1CCC(NC(=O)CC2CCC(C)(C)CC2)C1 CN1CCCc2ccc(NC(=O)Nc3cc(S(=O)(=O)CF)ccc3F)cc2C1 Cc1ncc(C(=O)NCC2CCCC2NC(=O)Cn2cccnc2=O)n1C N1(C(c2occ(C)c2)=O)CCCC(N(C(=O)C(N)=O)CC2CC2)C1 CC(C(=O)NC1CC(NC(C2COCC2(C)C)=O)C1)S(=O)(=O)c1ccc(F)cc1 c1(C(=O)OCC)ccccc1C(=O)NCCCNC(C1C=C(C)CS1)=O.CN N1(C(C2CCC(O)C2)=O)CCC2C(CCCN2C(C2CC23CCC3)=O)C1 Cc1ccc(CCn2nnnc2N(C)CC2CCC(C)(C)O2)cn1 CC1(C)CCCCC1CN1CCC(=CC(=O)Nc2ccccc2)CC1 c1(C(=O)NC2C(OC)CN(C(C(CC)F)=O)C2)cc2n(n1)CCNC2=O O=C1NC2(CCCC2)C2=C1C(c1ccc(I)c(Br)c1)NC(=O)N2CCF C1(CC(N2CCC(CCNC(C=CC)=O)C2)=O)(CO)CCOCC1 C1(C)(C(=O)NCC(CCOC)NC(=O)C(C)OC)CC2C=CC1C2 C1(OC)CN(C)C(C)(C(=O)N(CC(O)CN(C)C(C2CCCC23CCC3)=O)C)C1 C1(C)(C(=O)NC2CC(CCNC(c3c(C)cn(C)n3)=O)C2)CCOC12CC2(F)F Cc1onc(C(N2CCCC2C2(NC(=O)C=CC3CCCO3)CC2)=O)c1Br N1(C(C2(COC)CC=CC2)=O)CC2(C1)CN(C(=O)CCC1CC1CC1CC1)CCO2 C(=O)(CC(C(F)(F)F)N)N(C(C)(C)C)C.C(=O)(C(CC)CC(C)C)C(=O)COCP(C)(C)=O C1(CNC(c2ccccc2CO)=O)CN(C(c2cn(CCCF)nn2)=O)CCO1 c1(CN2CCN(S(=O)(=O)C(F)(F)F)C3C2C3)cc2cc(Br)ccc2[nH]1 N1(C(COCC=C)=O)CCC(NC(C2CC2(C)CC)=O)C1C(C)(C)C C1(C)(CC)CC(NC(=O)CNC(C2CCC2)=O)CN1C(=O)Nc1ccc(Cl)nc1 C(CC(C)(C)C(=O)N1CCC(N(C(=O)C(O)C2CC2)CCO)C1)SC CCCC(C)(C)C(=O)N1CCN(C(=O)CCc2nncs2)C(c2ccccn2)C1 C1(C(=O)NCC(CC)C#N)CC(NC(c2nc(C)oc2C)=O)C1(C)C C1(CNC(=O)OC(C)(C)C)C2CCCN(Cc3ccc(Br)cc3Br)C2CO1 N1(C(CCN(C(C2CC2(C)C(C)C)=O)C2CC2)=O)CC2CC(N)CC2C1.CCO N1(C(CCOCCNC(c2ccn(C(C)C)n2)=O)=O)CC(C)CC1C c1(CNC(N(C(C)CC(N)=O)C)=O)ccccc1OC1CCC1 C(C(C)(CC)C(=O)N(CCO)CCN(C)C)NC(c1c(CC)cns1)=O N1(C(C2(COC)CC2)=O)CCOC2(C1)CN(S(=O)(=O)c1cccc(F)c1)C2 C1(COC)CCCCC1C(=O)Oc1ncc(CCc2ccccc2)s1.C1(=O)CO1 c1(C(=O)NC(C(=O)NCC(CC)SC)C2CCCO2)ncncc1OC N1(C(C(COCC)C)=O)CCC(NC(=O)CCC2CCC2)CC(O)C1 c1(CCCC)ccc(C(C)C(=O)N(C(C)CNC(C2(C)CC2)=O)C)cc1 CC(C)C(C(=O)N1CCC(C(=O)NC2(CCO)CCCCC2)C1C)C1CCC1 c1(C(N2C(CNC(c3cc(C)no3)=O)CCC2)=O)c[nH]c2cccnc12 c1(OCCC(=O)NC(C)C(C)NC(=O)C=Cc2cn[nH]c2)cc(Cl)cc(Cl)c1 c1(C(=O)NCC=CCNC(=O)C2=CSCS2)ccc2c(c1)SCCN2 C1(C(=O)NCC2CCCC(CNC(C3(N(C)C)CCC3)=O)C2)CC2(C1)CC21CC1 c1(-n2cc(C3CCCN(C(Cc4c(C)nn(C)c4)=O)C3)nn2)ccc(F)c(F)c1 C1(C(N(CCOC)CCNC(C2(S(C)(=O)=O)CC2)=O)=O)CCn2cc(C)nc2C1 C(C(C(=O)N(C(C)CC)C)NC(c1cnn(C)c1)=O)OC C1(COC)(CNC(C2CCC(C)(F)CC2)=O)CCN(C(C2CCC(C)C2)=O)CC1 c1(C(N2CCN(C(CC3CC(C(=O)OC)C3)=O)C3C2C3)=O)cccc2nccn12 c1(-c2ccc(OC)cc2OC)nc2c(s1)CN(C(=O)COc1ccccc1)CC2 c1(OC)c(C(=O)NC(CNC(C2CC2c2ccccc2)=O)CO)cccc1Cl C(=O)(C1CCOc2ccc(Cl)cc21)N1CC(O)(CCNC(c2n(C)ncc2)=O)C1 Cc1cc(CC(=O)NCC2CC(NC(C34CC(C3)C4)=O)CCO2)ccc1F N1(C(C(CC)OC)=O)CCC(O)(CCNC(c2cn(C)nc2C(=O)OC)=O)C1 C=CC(F)(F)C(=O)N1CCOC(CCNC(c2cn(C(F)F)cn2)=O)C1 N1(C(c2c(C(C)=O)cn(C)n2)=O)CCCN(C(=O)COC2CCC2)C(C)C1 Cc1conc1CC(=O)NCC1CC(CNC(=O)CNC(=O)C(F)(F)F)CO1 C1(NC(c2[nH]nc(OC)c2Cl)=O)CC2CN(C(c3ccc(CSC)o3)=O)CC2C1 CC1(C)C(C(=O)NCCN2CCC(NC(=O)CCn3cccc3)CC2)C1(F)F C1(C(N(C)Cc2ncc(C)o2)=O)CC12CC(NC(c1ccccn1)=O)C2 C1(NC(c2cc(CCC)[nH]n2)=O)CC=C(C(=O)N2CC(C)C2)C1 C1(NC(c2c(C)[nH]cc2)=O)CCCCCC1NC(c1cc(O)cc(Br)c1)=O C1(C)(N(C(=O)C(CNC(=O)COCC(C)(C)C)N(C)C)C)CCC(O)CC1 C1(CN(C(CCSC)=O)C)CN(C(c2cncc(N(C)C)c2)=O)CCO1 C1(CNC(=O)CCOC(C)=O)CCN(C(C2(CC)CC=CC2)=O)C1 CCC(C)(C)CC(=O)N1CCC(C)C(NC(=O)C=CC2CCCO2)C1 Cc1cc(CC(=O)NCC2CC2C(=O)NC(C)CF)cs1 N1(C(=O)CC(F)(F)F)CCC2C(C1)CN2C(c1cnn(C2CCOC2)n1)=O C(=O)(C1CCc2cccc(F)c21)N(C(C)CNC(c1cc(Br)n(C)c1)=O)C c1(C(=O)OC)cc(SC)ccc1C.C12(CSC1)C(=O)N2 C1(NC(C=Cc2n(CC)ncc2)=O)CN(C(=O)CCOCC2CC2)CC12CC2 O=C(C1Cc2ccc(Cl)cc21)NCC12CC1CN(C(=O)CCC(F)F)C2 c1(OC)cccc2ccc(C(=O)N(CC(C)NC(C3(F)CC=CCC3)=O)C)nc12 C1(CC2CC(CCC(=O)N3CCC3)C2)CCCCN1C(=O)CN1CCCCCC1 N1(C(C(C)C(C)(F)F)=O)CC2CCCC(NC(c3cnc(O)n3C)=O)C2C1 C#CCC(C(=O)N1CCOCC1CCO)NC(c1oc(C)cc1C)=O C1(CN(C(=O)CCc2cnn(C)c2)C)CCCN1C(=O)CCCC1CCCO1 C1(CC)CN(C(=O)C(CCF)NC(=O)C2=C(C)CCC2)C(C)CO1 c1(CCCC)nc(C)c(C(N2CCC(NC(=O)CSC3CC3)C2)=O)c(O)n1 c1(OCC(C)C)cccc(C(=O)N(C(C)CNC(=O)C=C(Cl)Cl)C)c1 C(C(C)C)(C(O)C(=O)NCCC1(NC(C2CC2(C)C(F)F)=O)CCC1)OC C12(NCC3C(OC(C)(C)C)CCC3)CCC(C1)OC2C C1(NC(c2c(O)ccc(CC)c2)=O)CN(C(=O)C(C)OCCC=C)CC2(CC2)C1 C1(NC(C(=O)NC2C(N)C2)=O)CC2(CCCC2)C1 CCC(C)CCCCC(=O)N(CCCCCC(=O)NC1(C)CC(F)C1)C N1(C(C23CC(C)(C2)C3)=O)CCCC2(CCC(NC(=O)CCn3ccnn3)C2)C1 C#CCC(C)(C(=O)N=c1cc(C)n(C(C)C)[nH]1)NC(=O)CCn1cccc1 c1(CN(C)C)ccoc1C(=O)N(C)CC1CCN(C(C2CCC(C(N)=O)C2)=O)C1 C(=O)(CCCCCC(C)O)NC1C(NC(c2c(CC)c(C)sc2)=O)CCC1 N1(C(c2cncc(N)n2)=O)CCN(C(C2CC(F)(CO)C2)=O)C2CCC12 C1(NC(C2CN(CC)C(=O)C2)=O)CC2CN(c3nc(C(C)(C)C)ns3)CC2C1 CC1C(NC(c2cccc(F)n2)=O)CCN1C(=O)C(c1ccccc1Cl)(F)F CCC(C(=O)N(C1CCCC1C)C)NC(=O)Cc1scnc1C CC1CC(CNC(c2cnc(N)c(Cl)c2)=O)CCN1C(=O)Cc1cncc(F)c1 C1(C(=O)N(CCCCCO)C)(CC)CCCN(C(=O)C2=C(C)CCC2)C1 N1(CCc2ccc(C(N)=O)cc2)CCCS(=O)(=O)CC1C1CC1 Cc1cc(NC(C2CCN(C(=O)C(C)CC(F)F)CC2O)=O)cc(F)c1 c1(C(=O)NC2(CC(=O)NCCn3c(CC)nnc3)CCC2)ccc(C#N)[nH]1 C(=O)(N1OC2CCC1CC2)C1(NC(=O)CN2CC(=O)NC2=O)C(C)C1 c1(-n2cc(C(CC)NC(C(C)(C)C(=O)O)=O)nn2)c(C(F)(F)F)cccc1C c1(C(=O)NCCCCNC(c2cn(CCC=C)nn2)=O)[nH]c2c(c1C)CCCC2 N1(C(C(CC)SC)=O)CC2CCC(N(C)C(c3ccc(C)nc3C3CC3)=O)C2C1 C1(C)(CNC(C2(C(=O)OC)CC2C)=O)CCN(C(=O)C(N2C(=O)CCC2=O)C)C1 N#Cc1ccc(C2CC2NC(=O)C2=CCC2)cc1.C12(F)CC(C1)NC(=O)NC2 C(C)(CNC(c1ccc(O)c(N)n1)=O)(CC(C)C)NC(c1c(C)n[nH]c1C)=O N1(C(c2c(CC)n(C)nc2)=O)CCC(O)(CNC(c2ccc(Cl)cc2Cl)=O)CC1 C12(CC=C)CCN(C1)C(=O)c1cc(on1)C(=O)N2.c1(C(=O)NC)ccncc1CC c1(C2C(C(=O)NCC(C3CC3)NC(c3cscn3)=O)C2)ccc(Br)cn1 c1(C2CN(C(C(C)OC(CSc3n(CC=C)nnn3)=O)=O)C2)cccc(F)c1 c1(Sc2c(C(N3CCOCC3C3CC3)=O)nccc2)cccc(Cl)c1 O=C1NCC2(CN(C(=O)NC3(c4ccc(F)cc4F)CC3)C2)N1 CCC(C)(C)C(O)C(=O)NCC1CC(F)(CNC(=O)CCN2CCC(F)C2)C1 c1(NC(NCc2cc(NC)on2)=S)c(C)ccnc1C c1(C(=O)NCC(c2ccccc2)NC(C(C)(CO)OC)=O)ccc([N+](=O)[O-])[nH]1 c1(C(N(CC(=O)OC)CC#C)=O)nc(N(C)C)nc(=N)[nH]1.C1CCO1 c1(NC2CN(C)CC2O)ccc(S(=O)(=O)N2CCc3ccccc3C2)cn1 C(=O)(C(CC)C(=O)N1CC(NC(C2(C(C)(F)F)CCOCC2)=O)CC1C)OCC c1(C(N2C(CNC(c3cc(CCC)no3)=O)CC2)=O)cn(CC)nc1C(C)C CC1COCCN1Cc1nc(-c2ccccn2)no1 C(=O)(C(Cn1ccnn1)NC(C1CC(CO)CO1)=O)N(CC(C)C#N)C CCCCCC(=O)NCC(=O)N(C)CCN(C(=O)CC1CCCC1(F)F)C(C)C N1(C(C(C)OCC)=O)CCC(C(N2CC(C#N)C2)=O)C1CC N1(C(C23CC(C)(C2)C3)=O)CCC2CN(C(c3cc4ccccn4n3)=O)CCC12 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)CSCC(N)=O)C(NC(=O)C(C)C)C1 N1(C(C2C(CC)CCC2)=O)CC2(C1)CN(C(=O)CCc1cccc(F)c1)C2 CC(C)CC(O)C(=O)N1CCC2CC12C(N1CC2(CC=CC2)C1)=O C1(C(=O)NC2C=CC(C(=O)NC3(CC(F)F)CC3)C2)CCCC(F)(F)C1 c1(C(=O)NCC(CC(F)(F)F)NC(C2CCCC2CF)=O)coc2ccccc12 N1(C(COCCSC)=O)CC(NC(=O)CC2(C)CC2(Cl)Cl)C(c2nccn2C)C1 C1(NC(CS(N)(=O)=O)=O)COCCN(C(c2cccs2)=O)C1 c1(C(=O)NCC2C=CC(NC(c3c(C)nco3)=O)C2)ccc(F)c2[nH]ccc12 C1(C(=O)NC2CCN(C(C3(N(C)C)CCCC3)=O)C2)CCOCC12CCCCC2 c1(OC)cc(Cl)cc(CN2CCC(O)CC2C(N2CC(F)C(F)C2)=O)c1O CCN=C(NCCC1(CS(C)(=O)=O)CCC1)NCC1CC2CCC1O2 CCC(CC)C(C)C(=O)N1CCCN(C(c2cnc3c(c2)COC3)=O)C(C)C1 N1(CC)CC(C(=O)NCC2C(C)CCN2C(c2n[nH]c(C)n2)=O)CC1=O c1(C(N(C2CCN(C(C(C)(C)N(C)C)=O)C2)CC)=O)ccc(OC(C)(C)C)cc1 C1(OC)CCC(C(=O)NC2CC(CC(=O)NCc3[nH]cnc3C)C2(C)C)CC1 Cc1ccc(Br)c(NC(C2COCCN2C(=O)OC(C)(C)C)=O)c1F c1(C(CC(=O)NC(CO)CCCO)NC(CCC=C)=O)ccc(F)cc1F c1(C(N2CCNC(=O)C23CCC3)C(=O)NC(CC)C)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NCCC2(O)CN(C(c3cn(CC)nc3C)=O)C2)c(O)cccc1Cl C1(C(N2CC(N(C)C)C2)=O)CN(C(c2ccncc2OC(C)C)=O)CCS1 N12CCC3CC(C3C1)C2=O.c1(C(=O)N(C)Cc2nncn2C)ccc(S)cc1.CN c1(SCC(N2CC(C)C(NC(=O)COC3CC3)C2)=O)nc2ccccc2s1 c1(CC(=O)NCCN(C2CCCC2)C(C2C(CN(C)C)C2)=O)ccc(O)c(Cl)c1 C1(NC(c2cc(C)ncn2)=O)CC2CN(C(=O)Cc3cscn3)CC12 C(CC(=O)N1CCC(C#N)(CC)CC1)(CC(C)C)NC(C(C)NC(CC)=O)=O C1(O)(CNC(CCC(N)=O)=O)CCN(C(c2ccsc2)=O)CC1 C1(CC(=O)NC(C(=O)NCC(C(=O)OC)C)CC2CC2)OCCC1(C)C Cc1ncc(C(N2CCOC(C3CN(C(c4c[nH]nc4C)=O)C3)C2)=O)c(=N)[nH]1 [N-]=[N+]=NCCCCC(=O)NC(Cc1ccco1)C(=O)NCC(=O)NC=O c1(CCC(=O)NC2CCN(C(CSCC#C)=O)C2C(C)C)c(C)nn(C)c1C C1(NC(c2ccc(SCC)nc2)=O)CCCN(C(=O)C=Cc2cc[nH]n2)C1C c1(OCC(=O)NCCC2CN(C(C3C(C)(COC)C3)=O)C2)c(C)occc1=O C(=O)(C1=CCC(NC(C2(C)COC(=O)N2)=O)C1)N(C1CC(C(N)=O)C1)C C(CCC(=O)N(C(C)CNC(c1cnc(C2CC2)s1)=O)C)NC(=O)OCC C1(O)(CCNC(C2(C)CNC(=O)C2)=O)CCN(C(C2CCCCC2)=O)CC1 c1(-c2cn(C3CN(C(C(CN(C)C)O)=O)C3)nn2)ccc(N)cc1 C1(N2CCC(N(C)C3CC3)CC2)C2CCC1CN(C(=O)C=Cc1cccs1)C2 N1(C(CCC(C)OCC)=O)CC(C2CN(C(=O)C(C)CN(C)C)C2)C1 Oc1ncnc2c1CCN(N1CCCC(c3cccnc3)CC1)C2 c1(NC)cnc(C(N2CCC(CC(=O)N(CC#CCCO)CC3CC3)C2)=O)cn1 N1(c2nccc(OC)n2)CCC(C2CCN(C(C3CCC(F)(F)CC3)=O)CC2)C1 C(=O)(CC(C)CC(=O)OC)NCc1cn(CCCCC)nn1.C12CC1CNC2=O c1(C(=O)NC(C)C(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)cccc2ncn(C)c12 c1(N(C(=O)CCN(C(=O)CC2CC=CC2)C2CC2)C2CC2)c[nH]nc1Cl CCC(C)(C)C(O)C(=O)N1CC2(C1)CN(C(c1nnn(C)c1C)=O)C2 C(C)(C)(CC(F)C(=O)NC(C)C(C)(C)CN(C)C)NC(C(C(C)C)OC)=O C#CC1(O)CCN(C(C23CC(CO)(CN2C(c2c[nH]c(=NC)s2)=O)C3)=O)C1 C(=O)(C1=CCN(C(=O)CC2CC3CC3C2)CC1)NCC1(O)CCC(C)C1 N1(C(C2N(C(c3c(C)c(C#N)[nH]c3)=O)CC=C2)=O)CCC2(C1)CC2(F)F C(=O)(CC1=CCOCC1)NCCCC(C(=O)N1C(CN(C)C)C=CC1)O c1(C(=O)NC(C2CN(C(=O)C(CO)C(C)(C)C)CCO2)C)c(F)ccc(N)c1F c1(C(=O)NCC2CC(NC(C(CC=C)C)=O)CC2O)ncc(C)cc1Br C1(C(N(CC(C)SC)C)=O)C(C2CC2)CCN1C(C1CN(C)C1)=O c1(C(N2CC(C(C)NC(C(C(=C)Cl)(C)C)=O)OCC2)=O)ccc2c(c1)CC(=O)N2 C1(NC(=O)Nc2nccc(Sc3cccc(C)c3)n2)CC1C1CCCC1 N1(C(C(F)OC)=O)CCCC2(CCCCC2NC(c2nc(C3CC3)cs2)=O)C1 C1(CCC(=O)NCCC2CC(C(N(C(COC)C)C)=O)C2)CCC(=O)N1 c1(NCCC(CCC)C)cc(=NCc2cnc(C3CC3)nc2)[nH]cn1 Cc1cc(NC(=O)C(C)CN(C(=O)C(O)CC(C)C)C)cc(C)c1O CCCCC(O)CC(=O)N1CCC(CC)C1CNC(=O)COCCF N1(C(C=CC=CCC)=O)C2CCCC1CC(NC(c1cc(C#N)no1)=O)C2 c1(C(N(C)CC2N(C(c3c(C(CSC)=O)cco3)=O)CCC2)=O)cnncc1C c1(C(=O)NC(C)CN(C(=O)CCCc2nccs2)C)nnn2ccccc12 c1(C(C(=O)NCC(C)C)N(CC(CCC)C)C)ccc(F)c(C)c1 c1(C(=O)NCC(CNC(Cc2c(C)scc2)=O)(C)O)sccc1C#N C#CC1CCCN(C(=O)CC2CCN2C(=O)NC2CCC2C#N)CC1 c1(CN2C(C(N(C3CC3)CC)=O)CC2)cnc(OC)c(Cl)c1 C1(CC)CN(C(=O)CCN(C(=O)Cc2cn(C)cn2)C)CCN1C C(=O)(CC(O)CC(C)(C)C)N1CCC(C)(C(N2C3CN(C(C)C)C(C3)C2)=O)C1 C1(CNC(C2(C=C)CCC2)=O)CN(C(c2ccc(=O)n(C)c2)=O)CCC1C c1(OC)ccc(CCN(C(=O)C=CC(F)(F)F)CC)c(OCC2CCC(C)CC2)c1 CC1CC(NC(=O)Cc2ccc(Br)s2)CCN1C(c1cc(C#N)on1)=O CC1(CO)CCC(N=c2[nH]c(=NC3CCN4CCCC4C3)[nH]c3ccccc23)CC1 c1(C(=O)NCC2N(C(Cc3c(C)n[nH]c3)=O)CC(F)C2)ccc(C#N)nc1O C(=O)(C(CC)CCCCC)N1CCC(=C)CC1C(=O)N(C)CCOC c1(C(=O)NC2C(NC(C(C)C3CCCC3)=O)C2)cc(C(F)(F)F)cc(O)n1 C1(NC(CC2CC(=O)C2)=O)CCN(C(c2csc(Cl)n2)=O)CC12CCC2 C(CNC(=O)Cc1csnn1)(CC(F)(F)F)NC(C(N1CC(C)C1)C)=O C1(CC(=O)NCCC2(C(=O)NC(CC)C3CC3)CCCC2)CCN(C)CC1 N1(C(C(N2CCC(C)C2)=O)=O)CCN(C(c2cc(S(N)(=O)=O)co2)=O)CC(O)C1 C(CNC(c1ccnc(S)c1)=O)(CC(F)(F)F)NC(c1cccc(OC)n1)=O C123CC(C1)(C2(F)F)C(=O)NC1CC(C1)NC3=O.N1(C(=O)C2CC2)CCCC1 c1(CC2(C(=O)NCC(C)(C)N(CC(=O)OC3CC3)C)CC2)ccccc1 N1(C(CC(C)F)=O)CCC2CN(C(c3csc(-c4cnc[nH]4)n3)=O)CC12 C1(NC(C2(COC)CC(F)(F)C2)=O)CN(C(c2cn(C)cc2C)=O)C2(CCC2)C1 N1(C(=O)CC2CCCN(C(c3ccc(O)cc3)=O)CC2)CCC2(CCCC2)C1 Cc1cc(CC(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)ccc1Cl C(=O)(C#CC1(C(F)(F)F)CC1)NC(C(C)C)CCNC(C1NC(=O)C2CC12)=O CC1CCOC(C(=O)NCC2C(C)CCN2C(=O)CCNC(=O)CO)C1 c1(C(=O)NCC23OCCC(NC(c4n(C)cnc4)=O)(C2)C3)ccc(Cl)c(N)c1Cl CCCC(O)C(CO)NC(=O)CC1CC1CNC(=O)CCn1cnnn1 c1(CC)ccc(OCC(N2CCC(CF)(NC(c3cc(Cl)no3)=O)C2)=O)cc1 c1(C(N2C(CNC(CSCCC)=O)CCCC2)=O)cc(C)nc(O)n1 C(=O)(C1=CCCCC1C)NCC12C(CN(C(C3(CCC=C)CC3)=O)C1)C2 C(CCCC(=O)NC(CNC(C1CCCCC1C(F)(F)F)=O)CO)OCC CCN=c1ccc(C(N2CC(NC(C3(C)CCCC3O)=O)CC3(CC3)C2)=O)c[nH]1 C(c1ccc(S(C)(=O)=O)o1)=CC(=O)Nc1cccc(NC(C(CC#C)O)=O)c1 CN1CCC2CN(C(=O)NCc3nccn3CC(F)F)CC12 Cc1cc(C(N2CC(O)(CCNC(=O)Cc3cnnn3C)C2)=O)c(C)cn1 c1(C(N2CC(OC)(CNC(C3CCSC(C)C3)=O)C2)=O)cc2ccccn2n1 C(=O)(C1CC(O)c2ccccc21)N1CC(N(C(=O)CNC(=O)C(C)(C)C)C)C1 C1(C2CCN(C(=O)CC3CCC(=O)NC3=O)C2)(NC(c2c(C)coc2)=O)CC1 C12(C(N3CCC(NC(CSCC(C)=O)=O)C(F)C3)=O)CCOC1CCOC2 C1(C(N(CC(CC)NC(c2cc(OC)ccn2)=O)C)=O)CCN(C)C1=O N1(C(CCCCCC)=O)CC2CCCC2C1C(=O)N(CC(F)(F)CO)C C(=O)(C1CCCc2c1ncn2C)NCCCC1N(C(CCOCC)=O)CCCC1 N1(C(CCCCC#C)=O)CC2CCCC(C1)N2C(C1CCCCCC1)=O c1(OC)c(C(N2CCC2CNC(c2ccnc3[nH]ncc23)=O)=O)cc(Cl)cc1Cl c1(N(C(c2scc(C)c2C)C(=O)NCC2CCCO2)CC(=O)OC)ccccc1C N1(CC(=O)N(CC(N2CCOCC2)C)C)CCCC(C)(CNC(CO)C(=O)O)C1 CS(=O)CCC(=O)NC(C1CCOC1)CNC(c1scnc1C1CCCC1)=O c1(C(N(CC#C)C2CC2)=O)ccn(CCNC(=O)Cc2ccc[nH]2)c1 CCCCC(O)C(C)C(=O)NC(C)(C)C(C)CC(=O)NC(C)C(C)(C)C C1(CC(=O)NC(CC)CN(C)C(c2ccoc2CC(N)=O)=O)C(=O)ON=C1C C1(N(C(C(C2CN(C(C(C=C)C)=O)C2)OC)=O)C)CCOC(C)C1 c1(C(C(=O)NC2C(NC(C3CC4CC4C3)=O)CC2)CO)ccc(Cl)cc1 CC(C)S(=O)(=O)CC(=O)N1CCCC1CNC(=O)C=CCl c1(-n2ncc(C(=O)NC3CCC(CNC(CSCC#C)=O)C3)n2)ccc(Cl)cc1 N1(C(C2(COC)CCCO2)=O)CCC2(CCCN2C(c2cccnn2)=O)CC1 Cn1cc(S(C)(=O)=NC(=O)C2CC(=O)N(CSc3ccccn3)C2)cn1 Cc1cn2c(C(N3CCCCC(NC(C4(C)CC(F)C4)=O)C3)=O)c(Cl)nc2s1 C(=O)(C#CC1CCC2(CC1)OCCO2)N1CC(C)(NC(C(C)C(C)O)=O)C1 c1(C(=O)NCC2N(C(c3c(C)oc(C4CC4)n3)=O)CCC2)ncn2ccccc12 C(=O)(C1Cc2ccc(F)cc21)N(CC(C)(C)NC(C1CCc2nncn2C1)=O)C c1(CNC)ccc(S(=O)(=O)NC(=O)N(CCC2COC(C)(C)C2)C2CC2)cc1 c1(CNC(C(=O)OCC)Cc2ncccn2)n[nH]c2c1CCOC2 Cc1ccccc1C=CC(=O)NC1CCC1CNC(C1CC1C1CCCC1)=O C12(CNC(C3CC3(F)F)=O)CCC1CN(C(=O)C(O)Cc1cnc[nH]1)C2 c1(C(=O)NCCCN(C(=O)C(c2cnn(C)c2)C)CCC)cnc(O)cc1O c1(C2N(C(C(C(=O)NC3CC=CCC3)N(C)C)=O)CC2)ccc(F)c(F)c1 C1(C(N2CCCC(NC(c3c(CC)non3)=O)(CO)C2)=O)CCCC(C)(C)CC1 c1(CCNc2c(C)c(NCC3CCC(=O)N3)ncn2)cnc2n1CCOC2 c1(C(=O)NC2CCC(C)N(c3ncc(Cl)c(O)n3)C2)cc2cc(F)ccc2s1 CC1(CNC(C2CC(O)C2)=O)CCCN(C(=O)CC2CC3(CCO2)CC3)C1 C1(C(N(CC(CO)(CO)NC(C(C)OCC)=O)C)=O)COc2ccccc2O1 C1(NCC(C)O)CCN(C(C2(C)CC(Oc3ccncc3)C2)=O)CC1 c1(N2CCC(CSC)C2)ccc(S(=O)(=O)NC2CCC2c2ccccc2)cc1F c1(C(C)NC(C2CN(CC3CC4C=CC3C4)CC(=O)N2)=O)c(F)cc(F)cc1F c1(COC)nccc(N2CC3C(NC(c4cnon4)=O)C3C2)n1 N1(C(=O)OC(C)(C)C)CCOCC12CCN(C(=O)Nc1c[nH]c3ncccc13)C2 N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(C(N2CCCC2C#N)=O)C1 CC1CC(c2ccoc2)CCN1C(=O)NC(C)(C)C.C123CC1CCN2C3=O N1(C(CC=CC=C)=O)CCC2(CCOCC2)C(CNC(=O)Cn2[nH]cnc2=N)C1 C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)(OC)CCC12CCC2 C(CC1=CCCCCC1)NC(CC1OCCCN(C(C2=C(C)OCC2)=O)C1)=O C1(CC(=O)NCC(CC=C)NC(c2cnc(N(C)C)nc2)=O)COC(C)(C)C1 c1(CCC(=O)NCC2(F)CC(NC(=O)CC3CCC(=O)N3)C2)ccc(Cl)nc1 C1(C(=O)OC)CCCC1C(=O)N(CCCCNC(c1cnc(CC(C)C)[nH]1)=O)C c1(CC)c(C(=O)NCC2CC(COC)CN2C(=O)CC)nnn1CC.C(C)=O c1(N2CCC(C(=O)OCC)C2)nccc(Cl)c1[N+](=O)[O-] N1(C(c2c(C)[nH]c(C#N)c2)=O)CC(C(=O)NC(C)C(C)C)CC12CCC2 C(C)(N=c1nc(Cl)[nH]n2ccnc12)c1cc(OC)c(Br)cc1OC c1(SCC)cncc(N2CCCC2)n1.C1(C(N(C(C)(C)C2CC2)C)=O)CCCN1C(C)C C1(NC(c2ccc(C)nc2C)=O)CCN(C(c2cccnc2O)=O)CC(O)C1 Cc1cc(Br)ccc1S(=O)(=O)NC12CC(C(=O)N=c3cc(Cl)cn[nH]3)(C1)C2 N(C(=NCc1ccc(C(F)(F)F)cn1)N1CCC(CNC(=O)N(C)C)C1)C(C)C c1(C(=O)OC(C(=O)OC)COC(F)(F)F)ccc2nc(OC)ccc2c1 C1(C(=O)NC2(CC(=O)NC(C(CC)C)CN(C)C)CCC2)CCC(=O)N(C)C1 c1(C(=O)NC2C(C)N(C(c3nc(=N)cc[nH]3)=O)CCC2)cc([N+](=O)[O-])cnc1O Cn1c(S(=O)(=O)N2CCC3(CCNC3)C2)cnc1Cl CN1CCN(c2nnc(-c3cccnc3)s2)C(CNC(c2cc(F)cnc2O)=O)C1 N1(C(c2cnc(C)s2)C(=O)NC(CC)(C)C)CC(C)CC1(C)C c1(CC(=O)NCC2(O)CCN(C(c3nc(C)oc3)=O)C2)cncc2ccccc12 C1(NC(CNC(CC)=O)=O)CC2CCC(C1)N2C(=O)Cc1occc1C c1(CC)ccc(C(=O)NC(CCN(C(=O)C=Cc2cc[nH]n2)C)c2cccs2)[nH]1 Cc1ccc(O)c(CN2CC3CN(C(=O)Cc4cnc(N(C)C)c(F)c4)CC23)c1 C1(C(=O)NC(CCC)C)CN(C)CCN1C(=O)NC(C)C c1(C(N2C3CN(C(CC(C)(C)C(N)=O)=O)CC32)=O)ccc2ncoc2c1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)COCC3CC3)C2)=O)cc1)NC CC1CC(=O)NCC1C(N1CCN(C(C2CCC2(C)C)=O)C(CCO)C1)=O c1(C(=O)NC2CCCN(C(CCC(C)C)=O)C2C)cc(Cl)c(F)cc1F C(=O)(C(Cc1cnc[nH]1)N1CCC(OCc2cccs2)C1)NC(=O)OC(C)(C)C C1(C)(C(=O)NCC(C)NC(COCC)=O)Cc2ccccc2NC1=O C(=O)(C1=CCCCCC1)NCCCC1N(C(C(C)(Cl)Cl)=O)CCCC1 N1(C(c2ccc(CC)cn2)=O)CCN(C(=O)C(c2ccc(Cl)s2)C)C2CCC12 C1(C(=O)NCCn2cc(CNC(C=CCC)=O)nn2)CCC(=O)NC1 C12(C(=O)NCc3nccc(C(=O)NC4(COC)CC4)c3)C(=O)C3CC1C2C3.CO C1(NC(c2ccc(C)cc2)=O)CCCCN(Cc2ccc(O)c(C(=O)O)c2)C1 N1(C(c2c(C)ccnc2Cl)=O)CCC2(CC1)CC(C(=O)NC1CCCOC1)C2 N1(c2ncc(CCC)cn2)CCCC2(CCCN(Cc3ccc(O)cc3C)C2)C1 c1(CNC(C2(C=C)CCC2)=O)cnn2c1CN(C(c1cc(C)on1)=O)CC2 C(=O)(CCCCC)OC(C)(C)C.C=C(Br)CN(C1CN(C(C)=O)C1)CC c1(CNC(CC(=C)C)=O)nnc2n1CCN(C(c1cnc3sccn13)=O)C2 Cc1coc(C)c1C=CC(N1CC2(CC(NC(c3cnc(C#N)s3)=O)C2)C1)=O CC(C)CC(C(=O)NCC1CC2(CC2)C1)N(C)C(C1CC1C(F)(F)F)=O C(=O)(CC(C)C(C)(C)NC(=O)C(CC)CCOC)NCC1OCCN(CC)C1 N1(CCONC(c2ccncc2)=O)CCCC(N(C(=O)C(C)(C)CO)C(C)=O)C1.NCN c1(C(N2CCC(NC(CC3(C)CC3(Cl)Cl)=O)C2)=O)nc(O)nc(O)c1F C1(C(N2CC(O)(CCNC(=O)CC3CCCSC3)C2)=O)CCC(=O)N1C1CC1 C=C(C)CC(C(=O)N(CCCNC(c1cnc(OC)cn1)=O)C1CC1)NC(=O)NC c1(CC(N2CC(O)C(F)C2)=O)c(F)ccc2[nH]ccc12.c12csc(n1)NC(=O)C2 C(=O)(C(CC(F)F)c1ccccc1)N1CC(CNC(COCc2cc(C)on2)=O)C1 N1(C(C2(C#N)CCCO2)=O)CC2CC(C1)CN(C(=O)CCc1cc(Cl)cs1)C2 N1(c2snc(C(=O)OC)n2)CCC(NC(c2ccc3ncsc3c2)=O)C12CCC2 Cc1ccc2cc(C(N3CCC(c4nnc(S)n4C)CC3)=O)cnc2c1 c1(C(N2CCC(C)(NC(c3ccncc3)=O)C2)=O)cnc(Cl)c(N)c1 c1(C(=O)NC2CC(C)N(C(=O)CN(CC(C)(C)C)C)CC2)c(O)cc(F)cc1F N1(C(CC2(N(C)C)CC2)=O)CC2(CCC(O)CC2)C1.C1(CC=O)(C(=O)OC)CCC1 c1(-n2ncc(C(=O)NCC3N(C(COC4(C)CCCC4)=O)CC3)c2)ncc(Cl)cn1 Cn1cnn(CC(N2C(CNC(=O)CC3C=CCC3)CC3CC23)=O)c1=O C=CC(C)(CCOC)C(=O)NC1CCC1C(=O)Nc1cnn(C)c1CC C1(C)(C(=O)NCCCC(C)NC(CNC(=O)NC)=O)CCC2(CC1)CC2 C1(C(c2n(CCCC)nnn2)(C)NCC2CCC2(F)F)CC2CCC1CC2 O=C1CCc2cc(C(=O)NC3CN(Cc4cc(F)ccc4Cl)CC3F)ccc2N1 C1(C(=O)NCC23C(CN(C(C4(CC)COC4)=O)C2)C3)CC12CCOCC2 C1(C(=O)OC)CC2(C1)CC(C(N1CC(C)(CNC(C3C4CNC(=O)C34)=O)C1)=O)C2 N1(C(CC(C)(C(F)F)N(C)C)=O)CCC2(CCCCN(C(c3ccsc3)=O)C2)C1 c1(NC(c2nn(Cc3ccc(Cl)cc3)cc2Br)=O)cn2c(n1)CCC2 c1(N2CCC(CC(=O)Nc3cc([N+](=O)[O-])c[nH]3)C2)cc(Cl)nc(Cl)n1 N1(C(C2C(C)SCCC2)=O)CCC(C(=O)NCC2(O)CSC2)=C(F)C1 C(=O)(C1=CS(=O)CCC1)NC1C(CNC(C(C)CN(C)C)=O)COC1 c1(NC)ccc(C(=O)NC2CC(N(C)C(C3CC(C(F)(F)F)C3)=O)C2)c(Cl)c1 CCS(=O)(=O)c1ccc(CNC(=O)COc2ccc(CN=[N+]=[N-])cc2)s1 C1(NC(C(c2ccc(C)cc2)F)=O)CC(O)CN(C(=O)CCCN2CCCC2)C1 c1(C(=O)NC(CCCNC(COCC)=O)c2ccccc2)c2c(nn1C)CCC2 N1(C(C2CCC(CC)O2)=O)CCC2(C1)CN(C(C1CC=CCC1C)=O)C2 c1(CC)nc(C)sc1C(=O)N(C)CCOCCN(C(=O)Cc1ccccc1F)C c1(C(N2CCC(C(N3CC(CC)C3)=O)NC2=O)=O)nc(C2CC2)n2ccccc12 c1(C(=O)NC2CCC2CNC(C2CCCC(C(F)(F)F)C2)=O)ccccc1F c1(C(N2CC(C(=O)OC)CCC2C)C(=O)NCCCSCC)ccc(Br)c(O)n1 C1(NC(CC(=O)N(C)C)=O)(CO)CCCN(C(C2(C)CCCS2(=O)=O)=O)C1 O(P(=O)(CCC1CCCCO1)OSC)CC c1(C(N(C(CNC(C2CC(=O)NC2=O)=O)C2CC2)C)=O)cc(Cl)cc(Cl)c1F CC1(C)CCN(C(=O)C2=C(Cl)CCC2)CC1NC(=O)CC1CC1(Cl)Cl c1(C(=O)NC(C)C)ccc(NNC(=O)C(C)NCC(C)C)cc1 N1(C(c2ncn(C)c2)C(=O)NCCC2(C)CC2)CCCCCCCCCC1 C1(NC(C2C(c3n(C)cnn3)CC2)=O)CC2(CCN(C(C3CC4CC3C4)=O)C2)C1 n1(CC)nc(C)c(C(=O)NCC2CC(NC(=O)C3=CCCCO3)C2)c1C CC1CN(C(=O)CCC(=O)N(C)C)CCC1CNC(c1ncccc1F)=O C(=O)(C(C)(CO)NC(c1cccc(C)n1)=O)N(CCCC)CCO c1(NC(C(C)(C)CNC(c2cocn2)=O)=O)ccc(O)c(Cl)c1 C(=O)(C(CO)C(C)(C)C)N1CC(N(C(CN(CCC)C)=O)C)C(O)C1 N1(C(c2cnc(CCCC)s2)=O)CCOC(C)(CNC(C2(CO)CCCO2)=O)C1 CC(CCc1ccccc1)C(F)(F)CN=c1ccn(C2CCCCC2)[nH]1 CC1(C)CCCCCC1C(=O)NCCC1CSCCN1C(=O)Cc1cc[nH]n1 c1(C(=O)OCC)[nH]cc(C)c1C(=O)NC1CN(C(=O)CC2CCN(C)C2)CC1C CC1=C(C(=O)N2CCOC(CCNC(c3cncc(Cl)c3Cl)=O)C2)CCCO1 c1(C(=O)NCCN(C(C(C)SC)=O)CCCN(C)C)nc2ccccc2nc1O C1(Cc2onc(C)n2)CCC(N(CC2CCCC2)CC2CC2)CC1 C(N=C(NC1CCCCC1)N1CCC(OC2CC2)C1)c1c(OC)ncc(F)c1 Cc1ccc(C)c2[nH]c(C(=O)NCC(O)CNC(C34CC(C(C)C)(C3)C4)=O)cc12 C1(CNC(C2CCC(C)CC2)=O)CC2(CC2)CN1C(=O)COCc1ncnn1C C1(N(C(C(C2(O)CCC2)NC(c2ncn(C(C)C)n2)=O)=O)C)CCC(CO)CC1 c1(C(N2C(CNC(C(C(C)(C)C)NC(N)=O)=O)CCC2)=O)cc(F)c(F)cc1Cl C1(NC(CSC)=O)CCC(C)(CNC(c2cc(C(F)(F)F)cnc2O)=O)C1 N1(C(c2c(C)n(C)cc2)=O)CCC(C)C(CC(=O)NCC(C)(C)C2(O)CCC2)C1 Cc1cccn2ncc(C(=O)N(C(C)CCNC(=O)C=CC3CC3)C)c12 C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(C(CC#C)CC#C)=O)CC=C1 n1(CC(=O)NC2CC(N3CCNCC3)C2)ccc(C(=O)O)n1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2cscc2C2CC2)=O)CC1C C(CC(=O)NN=c1[nH]ccnc1N(C)C)n1cc(-c2scc(C)c2)nn1 C1(NC(C(C)n2cnnn2)=O)CCCC2CN(C(=O)C(O)CC(C)(C)C)CC12 c1(C(=O)Nc2nc(C(C)N)sc2)cncc(N=[N+]=[N-])c1 C1(CNC(C(C2CC2)OCC)=O)C2CN(C(c3cnc[nH]3)=O)CC12 c1(C(=O)OC)cc(NC(c2ccc(N3CCN(C)CC3)cc2)=O)cc(C2CC2)c1 c1(C(N2CC3CCN(Cc4cocn4)C3C2)=O)cc(I)ccc1[N+](=O)[O-] c1(CCNC(C2(COC)CN(C(=O)C(C)Cn3ccnc3)C2)=O)cccnc1O N1(C(CC(CC=C)NC(C2CCCCC2(C)C)=O)=O)CC2(CCC(=O)O2)C1 Cc1oc(C#N)cc1C(=O)NCC1(O)CCCN(C(=O)CC2CCCC2(F)F)C1 C1(C(=O)NCC(C(C)C)C)CCN(C(c2cc3n(n2)CCO3)=O)CC1C c1(C(=O)NC2CCN(C(c3c(C)noc3C)=O)C2)csc2c1CCC(C)C2 N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(=O)C=CC2CCOCC2)C2CC12 C1(NC(=O)NC(Cc2cccnc2)CO)COCC1C(=O)O c1(COC)cncc(N2CC(O)CC(NC(=O)CNC3CCSC3)C2)c1 Cc1cc(=O)n(CC(N2CC3CC(NC(=O)C(C)N4CCCC4)C3C2)=O)cn1 C(c1ccc2c(c1)NC(=O)CO2)=CC(=O)NCC(CC)NC(CSCCCC)=O c1(CC(=O)NC(CC)(C)CNC(c2ccsc2OC)=O)ccc2c(c1)CCCO2 CCCC(C(=O)NCC(F)(F)C(F)F)NC(c1cn(C)cn1)=O c1(C(N(C2CC(NC(C3N(CC)CCC3)=O)C2)C)=O)ccc(CO)c(Cl)c1 N1(C(CC2C(C(=O)OC)CC2)=O)CCCC1(C)CNC(=O)C=Cc1cn(C)cn1 C1(CNC(COCC=C)=O)(CO)CCCN(C(=O)C(C)P(C)(C)=O)C1 C1(C(=O)NCCc2ccc(CNC(=O)OC(C)(C)C)cc2)CCCCC12CCC2 C(=O)(C(CNC(=O)C(C)(C)n1cccn1)C(C)C)NCC(COC)C c1(COCC(=O)N(CC(C)NC(C=CC=CC)=O)C)ccc(C)cc1 C1(C(N2C(CNC(Cc3cc(C)n(C)n3)=O)CCC2)=O)CC(C)(C)CN1C N1(C(C(C)O)=O)CCCCC1CNC1CCCC1.c12ncc(s1)s2 Cc1cccc2ncnc(N3CC(NC(=O)C(c4cncn4C)O)CC3C)c12 C(CC(=O)O)(c1cccnc1)N(CC(=O)OCC)C.C1(=O)CCN1 c1(C(=O)NCCCN(C(=O)CN2CCCNC2=O)CC)cnn(CCO)c1N c1(C(N2CCC(CNC(c3cc(I)ccc3F)=O)CC2)=O)cc(Br)ccc1NC C(=O)(CC(F)(F)C(F)(F)F)N1CCC(N(C(C(=O)N(C)C)=O)C)C2(C1)CC2 C1(NC(Cc2c(C)nn(C)c2C)=O)CCC2CCN(C(c3ccc(Cl)[nH]3)=O)C1C2 c1(C(C(=O)NCCOC)N(C2CCN(C)CC2)C)cc2n(c1)CCCC2 N1(C(COC(C)(C)C)=O)C2CCC1CN(C(c1cncc(OC(F)F)c1)=O)C2 CC1(C)CN(C(c2coc(CO)c2)=O)C1C1CCN(C(c2ccc(Cl)cc2)=O)CC1 N1(C(C2C(C)CCO2)=O)CCC(C2CC2)C1C(=O)NCc1ccncc1 CC1CN(C(=O)C(C)(C)CC#N)CC(C)N(C(=O)C(C)NC(c2cccs2)=O)C1 c1(CN(CC(CNC(COC(C)=O)=O)O)C(=O)CC2(COC)CC2)ccc(C)cc1 CC1c2cc(Br)cc(Br)c2CCN1C(=O)N(CC1CCc2ccccc21)C N1(C(CCCC(=C)C)=O)CC(C2CN(C(=O)C(C)NC(N)=O)C2)C1 N1(C(c2scc(OC)c2)=O)CCC(CF)(NC(=O)C(F)C(C)C)C1 CC1Cc2cc(S(N)(=O)=O)ccc2N1C(=O)NCc1cc(Br)cc(F)c1F C1(C)(OC)CC(NC(=O)N(C(C)C)Cc2ccc(F)cc2)CC1(C)C CC1CCN(C(=O)CC2COCCO2)CC1CNC(c1ccc(OCF)cc1)=O C(C(C)(O)CN=c1[nH]cnc2c(F)ccc(F)c12)OC N1(CCCC)CCOCC1C(=O)NCC(C)NC(=O)CCc1ccc(C)s1 c1(C(N(CC(CC)NC(=O)C(C)(F)CC)CC)=O)cn(C)nc1C1CCOCC1 N1(C(C(=O)OCC(c2ccc(OC)c(OC)c2)=O)=O)C2CCCC1COC2 C1(OC)(CNCC23CC(c4ccccc4)(C2)C3)CN(C(C2CCCS2)=O)C1 c1(C(N2CCC(C)(CNC(=O)CSc3ccncc3)C2)=O)cnn2c1OCCC2 N1(C(C2C(C)(C)CCCC2)=O)CCC(CNC(=O)C2=CCCSC2)C(C2CC2)C1 C(=O)(C(O)CC(C)(C)C)N1CCCCC(C(=O)Nc2ccc(CN(C)C)cc2)C1 C#Cc1ccc(CCNC(N2CCN(c3cncnc3)C(=O)C2)=O)cc1 c1(C(N2C3CCN(C(c4c(C)ocn4)=O)C3CC2)=O)ccc2nc(Cl)ccc2c1 CC1CCC(NC(c2cnnn2C)=O)CN1C(c1nnsc1C(F)F)=O N1(C(C(CC)(C)O)=O)CCOC(C)(CNC(c2c(Cl)cncc2Cl)=O)C1 c1(C(=O)NCCC(C)N(C(=O)CC2CC3CCC2O3)C)cc(Cl)c(Br)[nH]1 c1(OCCCC)c(CCNCCC2(OCC)CCOC2)cc(Cl)cc1Br c1(OC)ccccc1Cn1cc(CNCC2CCC(C)N2C)nn1 C1(C)(C(N(C(c2cccn2C)Cc2ccc(F)cc2)C)=O)CCC(O)CC1 N1(CC)CCC(C(=O)OC)CC1.C12(CCCO1)C(=O)N1CCC1CC(=O)NC2 C1(CNC(=O)Cn2cnnc2)CC2CCCC2N1C(=O)CSC1CCS(=O)(=O)C1 c1(OC)ccc(C(=O)NCC2CC(C)N(C(c3ccccc3C)=O)C2)c(OC)c1 N1(C(CC(CC)CC)=O)CCN(C(=O)C(COC(C)C)NC(=O)OC)CC(O)C1 c1(OC)ccc2c(c1)C(NC(=O)C(N1CC3CC(O)CC1C3)=O)CCC2 c1(C(N2CCC(O)(C(CNC(CC(=C)Br)=O)C)C2)=O)c(C)ccc(C)c1N C(=O)(CC(C)(C)C(=O)NCC(CNC(=O)COc1cncc(Cl)n1)OC)OC C1(CNC(c2c(C)cc(Cl)cc2)=O)CC2CCCCC2N1C(C1CCC1)=O c12cncc(c1)C(=O)NC2=O.CCC(=O)N.C12(CC1)CNC2.C(=O)(C1CC1)OC c1(C(=O)NCC(CNC(c2cccc(C3CC3)c2)=O)O)cc(F)ccc1O c1(C(N2C3CC(C(=O)NCCCC(C)(C)CO)(OC3)C2)=O)cncc2[nH]ccc12 c1(NCCCS(=O)(=O)NC)nccc(=NCc2ccccc2CSCC)[nH]1 C1(OC)CCCC(CNC(=O)CSCCNC(c2nc(C)oc2C)=O)C1 Cc1nn(C)c(C)c1C(C)C(=O)N(CCN(C)CCn1cncn1)C(C)C c1(C(N(C2CC(NC(C3(C(F)F)CC(F)(F)C3)=O)C2)C)=O)cnc2n1CCC2 C1(NC(=O)C=C2CCCCC2)CCCC(NC(C(=O)NC2CC2)=O)C1 CS(=O)(=O)c1cc(C(=O)NC2CC2NC(=O)COCC2CC2)cs1 C(=O)(CCN(OC)C(=O)C1CCN(C(C2CC(C)(C)C2)=O)C1C)OCC CC1CN(C(C2(O)CCC2)=O)CC2(CCN(C(C3CCCOC3C)=O)C2)O1 C1(C(N2CCCC2CSC)=O)CC(F)CN1C(=O)OC(C)(C)C.C1(OCC)CCC1 C(=O)(C(O)C(CCC)NC(C1CCSC1)=O)NC1(C#C)CC(F)(F)C1 C=CC1CCN(C(=O)Cn2cc(CC3(CC(=O)O)SCCS3)nn2)C1 C1(CNC(C(C)(C)C)=O)CN(C(C2CCCCCC2)=O)CCC1C(F)(F)F N(C1CCc2cccnc21)C(C1CCN(C(C2C=CC=CC=C2)=O)C1)=O N1(CC(=O)N(c2cccc(C)c2)Cc2cn(C)nn2)CCCC2C(O)C(C)(C)C12 Cc1c(C(N2C(C(=O)NCC(F)CO)CC2C)=O)cccc1C#N C1(NC(=O)CC2CCCCC2)CCCC12CCN(C(c1cc(Br)cs1)=O)C2 c1(C(N(CCNC(c2sccc2-n2cnnn2)=O)CC)=O)csc([N+](=O)[O-])c1 Cc1ccc(CCC(=O)NC2CCC(NC(C3SCCCS3)=O)C2)cn1 C1(NC(C2(NC(C3C(OC)CCC3)=O)CCC2)=O)CCC(=O)NC1(C)C N1(C(c2cnc(C(=O)OCC)cn2)C(=O)NCCC)CCCNC(=O)C1C C1(NC(=O)CCCN2CCOCC2)CCCCN(C(=O)Cc2nccs2)C1 Cc1cc(N2CCOCC2CN(C(=O)C(O)CC2CCCCC2)C)n2ncnc2n1 CC12CCCCC1CN2C(C(=O)NC1CCC1)C1CC1 N1(C(COCc2cc(C)no2)=O)CCC(N(C)C(c2c(C)n[nH]c2C)=O)CC1 c1(OC)cc(C=CC(=O)NCCC(C)N(C)C(C2CCC(=O)O2)=O)ccc1F N1(C(C2CCCC(OC)C2)=O)CCN(C(=O)CCn2cnnn2)CC1CO c1(C(C)=O)ccc(C(N2CCCC2CN(C(=O)C(O)C2CCC2)C)=O)c(C)c1 C1(C(C(=O)NCc2cccs2)N(C)Cc2cn(CC)nc2)CCC2(CC1)CC2 N1(C(CC2CC(=C)C2)=O)CCOC(C(C)NC(=O)CSc2nncn2C)C1 C1(C(=O)NCC2C(NC(c3cn(C)nc3C(F)F)=O)C2)CCC2(CCC2)O1 c1(C(c2nnnn2C2COC2)NC(C)CCCCO)cc(Br)cc2c1OCC2 C1(C(=O)NC(C)CN2CCN(C)CC2)CC12CCN(C(c1cnns1)=O)CC2 N1(C(C(C)C2CC2)=O)CCC(C2(NC(c3cccn3C3CCCC3)=O)CC2)C1 Cc1cc(NC(C2CCN(CC(F)F)CC2)=O)ccc1NC(=O)CC(C)(C)F C1(NC(N(C2C(C)COCC2)C)=O)CC2(C1)CC(N)CCO2 c1(OCCOC)cccc(C(=O)NC2CC(CO)N(C(=O)CC(F)F)C2)c1 N1(Cc2nnnn2CC(F)(F)F)CCCN(C(=O)CC2CN(CC(C)C)C2)CC1 CC1CCC(NC(c2cn(C3CC3)cn2)=O)CN1C(=O)CCC(C)(C)C N1(C(C(CN(C)C)NC(CSCC#C)=O)=O)CC2CCC1C(O)C2O C1(NC(c2cncc(CC)c2)=O)CCCN(C(=O)Cc2ccnn2C)CC1 c1(C(=O)NCC(O)CCNC(C2(F)CCC2)=O)cnc2ccc(F)cn12 N1(C(C(CC)CC)=O)CC(CNC(c2ncc(F)cc2F)=O)C(C)(C)C1 N1(C(c2ncn(C)c(=O)c2)=O)CC2(C1)CN(C(c1csc(Cl)c1)=O)CC(C)(C)O2 N1(C(c2cc(C)n(C)n2)=O)C2CCC1C(NC(=O)CCOCC1CCCO1)C2 C1(C(=O)NCC2(CCNC(=O)C(O)c3ccsc3)CC2)CC12CCOCC2 CC(C)(C)C(CNC(C1CC2(CCC2O)C1)=O)C(=O)Nc1cnc(Cl)nc1 c1(C(=O)OCc2ccc(O)cc2)cnn2c1OCC2 N1(C(COCC)=O)CC2(CCCC(CNC(C3CC3c3ccccn3)=O)O2)C1 C(=O)(CC(C)CN(C)C)NCC(CC)NC(=O)CCc1ccc(C(C)C)cc1 C1(CNC(c2ccc(OCC#C)cc2)=O)CN(C(C2CCCN2C)=O)CC12CC2 c1(C(C(=O)NCC(C)NC(=O)C(O)CC2CCCCC2)C2CC2)ccccc1 C1(OC)CN(C(=O)CCCNC(=O)C(C)(C)C2CC2)CC12CC2 S(=O)(=O)(c1c[nH]ccc1=NCc1nc(Cl)cs1)N1CCCC(C)(CCC)C1 c1(C(=O)NCCC2CCCN(C(C(C)(C)SC)=O)C2)cnc(O)n(C)c1=O C1(OC)(CNC(c2ccc(F)cc2)=O)CCN(C(=O)C(c2cncn2C)(F)F)C1 Cc1csc2ncc(C(N3CC4CCN(C(=O)CC5CCCO5)C4C3)=O)c(=O)n12 C1(NC(Cc2n(C)ccc2)=O)CC2CCC1(C(=O)NCCCC(C)(C)O)C2 N1(C(c2ccc(C)c(Cl)c2Cl)=O)CC2COCC(C1)C2NC(=O)C(Cl)=CCl C(=O)(CC(C)CC(C)(C)C)N1CC(O)(C(C(=O)N(CCCO)CCC)F)C1 C=CCCC(C(=O)N(C(C)CN(C)C(=O)N)C)NC(=O)C=CCCC.NC c1(CNC(C2N(C(CC(CC)C)=O)CCSC2)=O)cccc(C#N)c1 C1(C(N(CCN(C(=O)C(C)C2CC2)C(C)C)C)=O)CCc2nncn2C1 Cc1cnc(CN2CC(C(N3CCCCC(C)C3)=O)CC(F)C2)c(F)c1 c1(C(N2C(C)CC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)coc2c(C)cccc12 CN1CCN(C(C2CCCN(C3CCC(=O)NC3)C2)=O)CC1 c1(C(=O)OCC)c(C)sc(CNCC2CCC(=O)NC2C)c1Cl N1(C(C2CC2C2CCC2)=O)CC2CCCC(C1)N2C(C1CCC2CC2CC1)=O c1(CC)cc(C(N2CC=CC2CNC(C2CN(C(=O)NC)C2)=O)=O)ns1 Cc1[nH]c2ccc(F)cc2c1C(N1CCCN(Cc2cnccn2)CC1)=O c1(C(=O)NC2CC(CCNC(C3C(CC(C)(C)C)C3)=O)C2)ccc(O)cc1O O=S(=O)(c1cccc(S(=O)(=O)N2CCCC2)c1)NC1C=C(c2ccccc2)C1 CC1CN(C(=O)CSCC(=O)OC(C)(C)C)CCC1NC(=O)CCc1ccc(Cl)s1 C1(CNC(c2c(OC)ccs2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC2(CCC2)O1 C1(CC(=O)OC)CCCCCC1.C(=O)(CC(=O)N)NC(COCCC(C)C)CO N#Cc1c(NC(C2CC(F)CN2Cc2cccc(O)c2Br)=O)cccc1F Cc1sc(C(N2CC(O)(C(C)NC(c3ccc(C4CC4)o3)=O)C2)=O)c(C)c1C c1(NC(CC)=O)ccc(C(=O)NC(=O)CCC(=O)c2ccccc2)cc1 C1(CCNC(C(C=C)O)=O)CSCCN1C(c1cc(Br)nn1C)=O N1(CC(=O)NC2(CNC(C3(C(=O)OCC)CCOC3)=O)CCC2)CCCC(C)C1 c1(C(=O)NC(C)CNC(=O)CC2(O)COC(C)(C)C2)ccc2c(c1)C(C)(C)CN2 C1(C(=O)NC(C(=O)NCc2ncncc2NC)COC)CC(C(C)C)=NO1.C(C)(C)O Cc1nc(C(=O)NC2CCC2NC(c2cc(Cl)c(F)cc2N)=O)c2ccccn12 Cn1c(C(=O)NCC2(C(N3CCCCC3CCO)=O)CC2)cnc1[N+](=O)[O-] C1(NC(C2CC(C)(F)C2)=O)CC2CCC1CN(C(c1cc(C#N)ccc1N)=O)C2 CC1C(NC(c2cnc(Cl)c(C3CC3)c2)=O)CCCN1C(C1CC2(CCC2)C1)=O C1(C(N2CCC(OC)C2)=O)C2CCCC1CN(Cc1ccc(F)cc1)C2 S(=O)(=O)(CCC(=O)OC)NC(c1n(CC)cnc1Cl)c1nnnn1CC c1(C(=O)NCC2C(NC(C3(C#C)CCCC3)=O)C2)cc2cc(Br)cn2cn1 CC(C)C(C(=O)NCc1ocnc1C(C)C)C(C)NC(=O)C=CC(=O)N(C)C CC1(C)CC(CNC(c2nnn3ccccc23)=O)CN(C(c2coc(Cl)c2)=O)C1 Cc1ccc(C)n1CC(N1CCCC(CNC(C2CC(=O)N(C(C)C)C2)=O)C1)=O C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(=O)C=C2CCCC2)C1 N1(C(C(C2CCCC2)NC(CC2ON=C(C)C2)=O)=O)CC(O)CC1C(N)=O c1(C(=O)NC(C(C2CCCCC2)NC(CSC)=O)C)ccc(C(=O)OC)cc1Cl C(=O)(CCCCCCOC1CCC(=O)C1)OCCC1(C)CCOC1 c1(OC(CC)C)ccccc1C(=O)NCC(O)CNC(=O)C(C)(C)c1cccs1 c1(C(N2C(CN(C(=O)CCCC(C)=O)CC)CCCC2)=O)n[nH]c2c1CCOC2 N1(C(c2c(CC)n(CC)nc2)=O)CC(C2(NC(c3c[nH]c(C(N)=O)c3)=O)CC2)C1 C(c1ccc(Br)cc1)=CCNCc1c(C)nccc1 c1(C(N2CCC(C)N(C(=O)C(=O)NCC(F)F)CC2)=O)cccc2c1C(C#N)C2 C#Cc1cccc(C(=O)NCC(C)CNC(c2cc(CCC3CCC3)c[nH]2)=O)c1F C(=O)(C(C)CNC(=O)C=CC(C)CC)NC(C#C)(C)C1CC1 CC1CCC(NCc2nc(C(F)(F)F)cs2)CN1C(=O)OC(C)(C)C C12CCN(CC1)C2=O.C1(C(N(CCOCC(=O)OC)C)=O)CCC1NC(C)C C12(C(=O)NCc3nccc(C)c3)CC(CO)(CN1C(C1CC3COCC3C1)=O)C2 C1(CNC(CC2(C)CC2)=O)(NC(C2(N=[N+]=[N-])CC2)=O)CCCC1 c1(NCC2CC(C)N(C(=O)Cc3ccccc3F)C2)cc2nncn2cn1 c1(OC)cccc(Cl)c1CNC(N1CCC(C)C(NC(=O)OC(C)(C)C)C1)=O C(=O)(CC(C)CN=C(NCC1(O)CCN(C)C1)NC1CCCCC1)OC C1(CC#C)(C(=O)NC23CC2CN(C(=O)CCc2cnc[nH]2)C3)CCCCO1 C1(NC(CC(C=C)(C)C)=O)CC2CN(C(c3sccc3NS(C)(=O)=O)=O)CC2C1 C1(NC2CC3(C(NC(Cc4cccc(OC)c4)=O)C3)C2)CC(C(=O)OC)=NO1 C1(NC(CC(C)C(F)F)=O)CN(C(=O)CCSCC(N)=O)C2(CCOCC2)C1 Cc1nc(C(N2CC(NC(c3ccccc3OC(F)(F)F)=O)C3CC23)=O)c(C)s1 c1(OC)cncc(CNC(=O)CN(C(c2nccnc2N)=O)C(C)C)n1 Cc1cc(NC(CCO)C2CC2)c(C)n1C(C)C(C)C C#Cc1ccc(C(N2CCCC2CS(C)(=O)=O)=O)cc1C N1(C(c2cnc(SC)n2C)=O)CCC(NC(C2CC2C)=O)C(F)C1 C1(CC(=O)N(C)Cc2ccc(CC)o2)CN(C(=O)C=CC(F)(F)F)CCC1C C(=O)(C(F)C(=O)N1CCN(CC(C)NC(=O)CCc2ccnn2C)CC1)OCC Cn1cc(Cl)c(C(=O)NC2CCCCC2NC(=O)C(O)CC2CC2)n1 C1(NC(c2sccc2F)=O)C2CC1CN(C(C1COCCC1(F)F)=O)C2 CN=c1[nH]cc(C(=O)NCc2cc(C(N3CCOC(C(C)C)C3)=O)n(C)n2)s1 c1(CN(C2C(NC(c3cc(OC)n[nH]3)=O)CCCC2)C)nc(Cl)nc2[nH]cnc12 c1(NC(C2(F)CN(Cc3cccc(C#N)n3)C2)=O)cccc2c(Cl)ccnc12 c1(C(=O)NC(C)C(C)(C)NC(=O)C2=CCCC2)cc2ccnn2cn1 c1(C(=O)N(C2(CC(N3CCC(OCC(N)=O)C3)=O)CCC2)C2CC2)cnncc1O c1(OC)ccc(CN2CC(C)(CNC(=O)COC3CCOC3)C2)c([N+](=O)[O-])c1 Cc1cc(C(=O)NCC23CC2CN(C(=O)C#CC2CC2)C3)ccc1F C1(NC(CN(C)CC)=O)(CO)CCCN(C(=O)C(C)CSC)C1 C1(C)(CNC(CC2CCCC(C)O2)=O)CC(F)(F)CN1C(c1cnn[nH]1)=O CCC(C)C(O)CC(=O)NC1CCOC1C(=O)NCC(C)(C)C1=CCCC1 C1(F)(NC(N2CCC(C(C)C(=O)Nc3cnccc3Cl)CC2)=O)CCCC=C1F Cc1ccc(S(=O)(=O)N2CCCC(CC(=O)Nc3cncnc3O)C2)cn1 C1(C(=O)NCCOCCOCC#C)CC(O)CCN1C(=O)C(CC)OCC Cn1nnc2cc(C(=O)NC3COCCC3NC(c3cccc(C4CC4)c3)=O)sc12 N1(C(Cc2c(C)cco2)=O)CCC(CO)(NC(C2CC23CC3)=O)CC1 C(CNC(c1ccccc1)C)(C(C)C)OC.C1CCS1 c1(OCC)cc(NCC2(OC)CCCC2)nc(C)n1.C12CCCCC1NC(=O)C2 Cc1nc(Br)ccc1-n1nc(CCO)nc1C1CCCOCC1 C(=O)(CC(F)(F)CS(C)(=O)=O)NCC(CCOC)NC(c1cc(C(N)=O)c[nH]1)=O c1(CC(=O)NC(CNC(C2N(CC)CCC2)=O)(C)C2CC2)nc2ccccc2s1 Cc1cc(N2CCC(CNC(=O)CCCC3CC3)C(C)C2)nc(Cl)n1 C1(NC(C2C(CNC(c3cncc(COC)c3)=O)CC2)=O)CCN(C)C(=O)C1 c1(C(N2CCN(C(CC(CCC)C)=O)CC2CCO)=O)cc(F)c(C#N)c(F)c1 C1(NC(C(CCC)OC)=O)CN(C(=O)CCCn2cncn2)CCC12CCC2 CC(C)CCC(F)C(=O)NCC(CC1CC1)C(=O)NCCCn1cnnn1 c1(C(=O)NC2C(CNC(=O)Cc3cncn3C3CC3)CC2)n[nH]c2c1CCOC2 N1(C(c2c(CC#N)ccs2)=O)C2CCC1CC(NC(C1C=CCC1)=O)C2 Cc1cccc2cc(C(=O)N(CCCOCCNC(=O)CC3CC3(C)C)C)oc12 CC(C)CC(C)(C)C(=O)NC1CCCC1NC(c1ccccc1CO)=O C1(NC(CC(C)F)=O)CCC(NC(c2nccnc2N)=O)CC1 C(=O)(C(C)CO)N(C(C(=O)NCCOC(C)C)C1CC1)C CN1CCN(S(=O)(=O)CC(=O)NCC(C2CCC2)CC)CC1.C(=O)(C(N)=O)C.C(=O)N CCCC(CC1CCCC1)C(=O)NC(C)(CNC(=O)C(C)(C)CO)C(C)C C1(NC(C(CC=C)OC)=O)COC2(C1)CN(C(=O)CC1OCCO1)C2 c1(C2(SCC3CCCN(C(c4cccc(OC)c4)=O)C3)CC2)cc(C)ccc1F N1(C(C2(C)CCC(C)CC2)=O)CC2CC(C1)CN(C(C1CN3CCN1CC3)=O)C2 c1(C(N2CC(NC(C3C(CCC)CCC3)=O)(CO)C2)=O)cnc2c(c1)COCC2 c1(OC)ccccc1C(CNC(=O)C(C)CO)NC(=O)CSc1scnc1C C1(C(=O)NCCCC(C)O)CN(C(=O)C2=CCSC2)CC1(C)C c1(NC(=O)C(N2CCC(CNc3ccco3)C2)=O)ccc(F)c(I)c1 C1(NC(C2(CCOC)CCC2)=O)CCC(C)(CNC(=O)CC(F)F)C1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CN(C(=O)C(O)CC(F)F)C2(CCC2)C1 N(C1CCCc2occc21)C(C(N(C(C(=CC1CCCC1)C)=O)C)C1CC1)=O C1(C2CCCN(C(c3ccnc(C)c3Cl)=O)C2)(NC(CN(C2CC2)CC)=O)CC1 c1(OC)ccc(COC(=O)C(c2ccccc2)NC(=O)COC2CCCC2)cc1 C1(NC(C2CCCNC2=O)=O)CC=CCC1C(=O)NN1CC(F)CC1c1nc[nH]n1 C=C1CCN(C(=O)OCC)C(C(=O)NC2COCO2)C1 N1(C(CCc2c(C)nc[nH]2)=O)CC2(CCOCC2)C1c1cnn(C)c1 c1(C(=O)NCC(CC=C)NC(=O)CCCc2nc(C)no2)cc2c(s1)CCC2 N1(C(c2ccc(OC)o2)=O)CC(C)(CNC(=O)C(C2CCOCC2)O)CC1(C)C c1(C(=O)NCCN(C(C(n2c(C)ccn2)C)=O)C(C)C)cnc(=NCCF)[nH]c1 C1(NC(CC(COC)C)=O)CCC2CN(C(=O)C(=O)Nc3ccccc3)CC2C1 c1(C(=O)NC(CNC(C=C(C)c2cnn(C)c2)=O)(C)CO)ccc(S(C)(=O)=O)s1 c1(C(=O)NC(C2CCCN(Cc3nnc(S(C)(=O)=O)s3)C2)C)c([N+](=O)[O-])cnn1C C(=O)(C1=CS(=O)CCC1)N1CC(C)C(CNC(C2(C)CNC(=O)C2)=O)C1 C1(NC(C)CCO)COC2(CCN(c3ncc4[nH]ccc4n3)CC2)C1 C1(NC(C2CC(OC)C2)=O)CC2CCCC(C1)N2C(c1ccc2nccn2c1)=O N1(C(C2C(CC)OCC2)=O)CCOC(C)(CNC(C23CC(C)(CO2)C3)=O)C1 CCC(C)(C)CC(=O)N1CCOCC(CNC(c2c(Cl)nsc2Cl)=O)C1 CCCC(CNC(c1cc(C)nn1C)=O)C(=O)NC1CC12CC(OC)C2 C1(C(=O)NC(CC)CO)(CO)CCCN1C(=O)OC(C)(C)C Cc1nc(C(=O)NCC2(C(=O)NCCN3CCNC3=O)CC3(CC3)C2)c(C)s1 c1(C(N2CC(NC(c3n(C)cnc3)=O)C(F)C2)=O)cc2nnn(C)c2s1 CN1N=C(C(=O)N2CCC3CCN(C(c4ccc(=N)[nH]c4Cl)=O)C3C2)CCC1=O c1(C(N2CC3CC3C2)=O)cnc2ccc(C3=CCC(O)CC3)cc2c1Cl C(CC(=O)N1CC(O)CCO1)C1N(C(=O)Cc2ccccn2)CCC1 c1(CC(C)C(=O)N2CC(O)(CCNC(C3C(F)(F)C34CC4)=O)C2)ccccc1Cl c1(OC)ccc(S(=O)(=O)N2CCCC(C(=O)C3CC3)C2)cc1.C12C=CCCN1C2 Cc1ncc(S(N)(=O)=O)cc1C(=O)NCC(F)CNC(C1CCC(C)O1)=O c1(OC)ncc(CN2CCC(C(=O)NC(C)(CO)CO)C(O)C2)cc1Cl C(CCC(C(=O)NCCc1cocn1)NC(c1cc(CO)on1)=O)OC C(=O)(C1=CCN(C(=O)Cn2c(C)cnc2O)CC1)NC(CC)CC CC1CC2CC2CC1C(=O)NC.c12ccc(cc1)CC1C(CCC1)NC(=O)C2 S(=O)(=O)(c1ccc(Br)cc1F)Nc1ccc(C(C)(C)C)o1.C12CCCN(C1)C2 c1(C(N2CCC(NC(C3CCC(C#N)CC3)=O)CC2)=O)ccn2cccc2c1 N1(CC(=O)NCC(C)(C)OCCNC(C2C(C)CC2C)=O)CCC(=O)NC1=O C12(C(=O)NCc3c(C)noc3C)C(NC(c3ncc(F)cc3F)=O)C3CC1C2C3 CCCC(F)(F)C(=O)NC1(CNC(c2cn(C)nc2COCC)=O)CC1 C1(CC(=O)N(C2CCN(C(=O)C(C)C(=O)OCC)C2)CCC)(SC)CCCCC1 c1(C(=O)NC(Cn2cc(C(C)OCC)nn2)C)ccc2c(Br)cnn2c1 c1(NC(CN(CCNC(C2N(CC)CC2)=O)CC)=O)cnsc1C C#Cc1cc(C(=O)NCC(C)(O)CNC(=O)C(C)(C)N(C)C)cc(F)c1 C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCC#CCNC(C(C)OCCCC)=O C1(C(=O)NCC2CC(NC(c3c(C(=O)OC)c[nH]c3)=O)C2)CCN(C)C1C c1(CC(=O)NC2(CNC(C(CC)O)=O)CCOCC2)cc(F)c(F)cc1F CC(C(=O)NCC(C1CC1)NC(C1CC(=O)C1)=O)S(C)(=O)=O C(=O)(CCCCCSC)N(C)CC1N(C(C2CCCN(C(=O)OC)C2)=O)CCC1 c1(C(N2CC(NC(=O)C(C)CC3CC3)CC(OC)C2)=O)n[nH]c2c1CCOC2 C1(C(=O)NCC=CCNC(C2(OCC)CCCCC2)=O)CCn2ncnc2C1 c1(-n2cc(C(C3N(CCOC)CCC3)Sc3ccccc3)nn2)ccccc1F c1(C(C(=O)NCCCSC)N(c2nccs2)C)cn2cccc(F)c2n1 Cc1cc(C(=O)NC2CCC(C)(N3CCOCC3)CC2)nnc1O c1(SCC(=O)NCC2CCCC(NC(C(C)CF)=O)C2)nc2ccccc2n1C C1(CCNC(C2CC3CC2C3)=O)CN(C(C2(c3ccccc3)CCC2)=O)CCO1 N1(C(CC=CC=C)=O)CCCC(C)(C)C1CNC(C1CCC(C)(C)OC1)=O Cc1nsc(N)c1C(N1CCC(C(C)NC(=O)C#CC2CC2)CC1)=O C(=O)(C(C)(C)CCCO)N(C1CCCN(C(C2CC(CCC)OCC2)=O)C1)CC Cc1ccc(Cl)c(F)c1-c1cn(C2CC(C(C)C)C3OCCC23)nn1 N1(C(c2cnn(C)c2N)=O)CC2(CC(NC(c3noc4c3CCCC4)=O)CO2)C1 c1(C(=O)C2CC2)cc(C)on1.C1(C(CO)NC(COCCN)=O)CCCO1 c1(C(=O)NCCC2CN(C(CN(C)C)=O)C2)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 C=CCCCC(C(=O)N1CCC(F)(C(N)=O)C1)NC(=O)C(C)C(O)C(C)C Cc1nc(O)c2cc(C(N3CC(NC(C4CC5CCC4O5)=O)C3)=O)ccc2n1 C(C(CC(F)(F)F)NC(C1CCC1(C)C)=O)NC(C1(CC#C)CCC1)=O N1(C(c2c(F)ncc(OC)c2)=O)CC2CCC1CC2NC(C1(Br)CC1)=O c1(C(N(C2CCN(C(=O)Cn3nccn3)CC2)C)=O)cc(C(F)(F)F)cc(O)c1 CCCCCC(O)CC(=O)N(CCC(=O)NCCCCCCO)CC n1(CC(=O)NCCC2(NC(c3cc(C)no3)=O)CCC2)nc(C)c2c1CCCC2 CCCCC(CC)CC(=O)NCCN(CCOC)C(c1cc(Cl)nn1C)=O Cc1ccc(C(=O)NC2CC(NC(=O)CC3CC3C)C2)s1 C(=O)(C(F)(CNC(=O)C(C)(C)C(C)O)C(C)C)NCC1(C=C)CCC1 C1(CCNC(C(C)c2ccsc2)=O)CN(C(c2cn(C)cn2)=O)CC1C C(CCCCCC(=O)N(C)Cc1ccoc1C)NC(CC(C(=C)C)OCC)=O C1(C(=O)NC(C(=O)NCc2ccc(CC)s2)CO)CCCCC1O c1(C(N2CCC(C(C)NC(c3n[nH]cc3Cl)=O)C2)=O)ccncc1N1CCCC1 C12CN(C3(CCOCC3)C1)C2=O.Cc1nc(CN)oc1-c1ccccc1F C1(C(=O)Nc2cccc(N(C)C)c2)C(C2CC2)CCN1C(C1C=CC=CC=C1)=O CCCC(CC(=O)NC(C)COCC)NC(=O)CC1CCC(=O)NC1 CCCC(CCC)CC(=O)NC1(C)CC(NC(=O)C(F)(F)c2cccnc2)C1 C(=O)(C1CCc2c[nH]nc21)NCC(CCOC)NC(c1ccc(F)c(C)c1)=O N1(C(=O)NCc2ccncc2)CCC(F)(Cc2ccccc2)C1 CC(CS(C)=O)C(=O)NCC1CN(C(c2cccc(CN3CCOCC3)c2)=O)C1 c1(C(=O)NCCCC(C)NC(=O)C(C)(C)F)cccc(C(=O)OC(C)(C)C)c1 c1(C(=O)NCC2CCC(NC(c3c(C)ncs3)=O)C2)nc(O)c(C)s1 N1(C(CNC(CCCCC)=O)=O)CCC(NC(c2ccoc2)=O)C2(CCC2)C1 C1(C#N)(C(N(CC(=O)NC2CCN(CCC)C2)CCC)=O)CCCO1 C(=O)(C1CCc2ccc(OC)cc21)NC(C)CS.CCCOCCNC(C)=O n1(CC(=O)Nc2ccc(=O)n(Cc3cccc(Cl)c3)c2)cc(Cl)cc(I)c1=O Cn1[nH]c(C(=O)NC2(CNC(=O)CC3CC(CF)C3)CC2)nc1=O N1(C(c2nc(C)n(C)n2)=O)CCC(NC(c2ccco2)=O)CC(O)C1 C1(C(N2CCC(NC(C=CCNC(=O)C3CC3)=O)C2)=O)CCC2(CC2)C1 CC1(C)C=C(C(=O)NC2CC2NC(C2CCC(C)(C)OC2)=O)C1.CC=O N1(C(c2c(OC)csc2)=O)CCC(O)C(C(N2CCCCC2C)=O)C1 c1(OC)ccc2[nH]c3c(c2c1)CCN3C(=O)C(C)Oc1ccc(Cl)cc1C c1(-n2cc(C(CCC(C)=O)(C)C)nn2)cc(C(=O)NCCN(C)C)c(=O)n(C)c1 C1(C)(NC(C2CCC(C)O2)=O)CCN(C(=O)CC(C)F)CC1 C1(NC(c2c(C)onc2-c2ccccc2Cl)=O)CCN(C(=O)C(C)C)CC1F N1(C(C(C)=C(C)C)=O)Cc2ccccc2CC1CNC(=O)CC1CNC(=O)C1 C(=O)(C(C)S(N)(=O)=O)NCC1CCC(n2cc(-c3c(OC)nsc3)nn2)CC1 n1(CC(c2ccccc2)NC(CN(CCCC)C(C)=O)=O)c(C)ccc1C c1(CC)ccc(C(=O)OC)cc1NC(=O)C(=O)NC1CCN(C)C1C C(=O)(C1=CCC(C(F)(F)F)OC1)N(CCN(C(C1CCCCN1C)=O)CC)CC C=CC(C)CC(=O)NCC(C1CCCCC1)NC(c1cc(C(C)(F)F)on1)=O C1(CN(C(C2CCCC2F)=O)CC)CCCCN1C(=O)CCSCC(N)=O C(=O)(C1=CCCC1C)NCC(C)NC(c1cn(C)nc1Cl)=O CC(F)(F)CC(=O)NC1CCC(CNC(c2ccc(N(C)C)cn2)=O)CC1 S(=O)(=O)(c1cccc(S(=O)(=O)NCC(=C)CC)c1)NC(C)=O c1(C(=O)NC2(CNC(C3C(C(C)C)(CC)C3)=O)CC2)cc(O)cc(O)n1 N1(C(C2CCCOCC2)C(=O)NCC(=C)C)Cc2scc(Br)c2C1 c1(C(=O)N(C2CC(OC)CN(C(C(F)(F)OCC)=O)C2)CC)ccc2ncsc2c1 N1CC2(CNC(=O)N2C)C1.C(=O)(C1=C(C)OCCO1)N1CCN(CC(=O)NC)CC1 c1(C(=O)CN2CCNCC2)cc(F)ccc1[N+](=O)[O-].C(CCF)N1CCC1 c1(C(N2CC(F)CC(C(=O)NC(C)(C)CO)C2)=O)cc(F)c2cc[nH]c2c1 C1(N(C(=O)CNC(=O)CNC(=O)CC(C)n2cccn2)CC)C2CC(=O)CC12 N1(C(c2nc(C(C)OC)oc2)=O)CCCC(O)(CCNC(c2cnns2)=O)C1 N1(C(c2c(Cl)cc(C)s2)=O)CCN(C(C2CCS(=O)(=O)C2(C)C)=O)CC(CO)C1 N1(C(C=C(C)C)=O)CC2CCC1CC2NC(=O)CC(C)(C)O N1(C(c2nc(CCC)oc2)=O)CC(NC(C2CCC=CO2)=O)CC2(CC2)C1 c1(C(=O)NCCCC(C)NC(C2CC3C=CC2C3)=O)cnn2cc(C#N)cnc12 N1(C(c2cn(C)nc2)=O)CC(CNC(=O)Cc2cccc(OCC#N)n2)C(O)C1 C1(C(N(CC(C)C#N)C)=O)CC2CC1CC2NC(=O)CCC(N)=O n1(CC(=O)NC2CN(C(c3ccc(C)cn3)=O)C(C)(C)C2)cc([N+](=O)[O-])c(C)n1 C=CC(CC)C(=O)NC(C1CCN(C(C2CC(OC(C)(C)C)C2)=O)CC1)C Cc1cccc2oc(C(=O)N(C)CC3CCCN(C(=O)CC4CC(F)C4)C3)cc12 c1(OC(C)C(=O)NC2CCC(NC(=O)CCN3CCCC3)C2)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(C)CNC(c2ccnn2CC(F)F)=O)cccc(Br)c1 N1(C(C(CN(C(=O)C(O)C2CC2Cl)C)(C)C)=O)CCCN(C)C(=O)C1 N1(C(=O)Cc2ccno2)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C2(CCC2)C1 N1(C(C2(CC)CCOC2)=O)CCCC2(CCCN2C(c2cnn(C)c2C)=O)C1 C(CCCCCN(C(=O)CC1CC(F)C1)C)NC(C(C)NC(CC)=O)=O Cc1cccc(CCC(=O)NCC2CCCOC2c2ccccc2)n1 Cc1ccc(C(=O)NC2CC(C)CN(Cc3ccnc(F)c3)C2)cc1Cl C1(C(N(C2CCCOC2)CC)=O)COC(CNC(=O)CCCOC(C)=O)C1 C#Cc1c[nH]nc1C(N1CCCC1CN(C(=O)Cc1cn(C)nc1C)C)=O C(=O)(CS(=O)(=O)C(C)C)NCC1C(CNC(C2(OC)CCCCC2)=O)C1 c1(C(=O)NC2COC3CN(C(COCC)=O)CC32)cnc(O)c2cccnc12 CC(C)C(C)CC(=O)NCC1C=CCN1C(=O)C(O)CCN(C)C n1(CC)nc(C)c(C(=O)N(CC(C)N(C)C(=O)Nc2n[nH]c(Cl)c2Cl)C)c1C C(=O)(C(CC(F)(F)F)NC(=O)Nc1cccnc1OC)OCCCC C(=O)(CC(F)(F)F)NCC(CC=C)NC(c1nccnc1OC)=O n1(COC(c2ncnc3c2ncn3CCl)=O)c2ccccc2c(=O)c2ccccc12 C(CCN=C(NCC1CCC(O)C1)N1CCC(F)C1)OC(C)C c1(C(=O)NC2C(NC(=O)Cc3cccnc3)CCC2)cnc2c(F)cccc2c1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC2(CNC(c2csc(C)n2)=O)C1 C1(C(N(CCOCCNC(c2c(CC)c[nH]n2)=O)C)=O)C(O)C(=O)N(C)C1C C12(C(N(C(C#C)C)C)=O)CC(NC(C3CCCSC3)=O)(C1)C2 c1(CC(=O)NCCN(C(=O)C2=NOCC2)CC)cc(C(F)(F)F)cc(Cl)n1 CCCCC(C)C(=O)N1CCCC1C(C)(C)NC(=O)CCc1nc[nH]n1 N1(CC(=O)NC(C)(C)CNC(c2cnn(CC3CC3)c2)=O)CCCCCC1 c1(CNC(C(C2OCCO2)OC)=O)cnccc1C n1(CC(N)=O)cc(C(=O)N(O)Cc2cn(CC3CNC(=O)O3)nn2)nn1 CCC(CN(C)C)CC(=O)N(CCC(=O)N1CCS(=O)C(C)C1)OC C(=O)(C1=NOC(c2ccccc2)C1)NCCN(C(C)C)C(C1CCCN(C)C1)=O Cc1nc2ncnn2c(C)c1CC(=O)NC1CN(C(c2ccoc2)=O)CC12CC2 c1(C(N2CCC(OCCNC(c3c[nH]nc3F)=O)C2)=O)ccc2c(c1)OCO2 C1(NC(c2ccnnc2)=O)CN(C(=O)Cc2ccc(Br)s2)CCC1CO C1(C(=O)O)(NC(c2cnc(-c3ncccn3)s2)=O)CCNCC1 c1(N(C)C)cccnc1N(C)C(c1ccc(NC=O)cc1)=O.C1C(O)CN1C C(c1ccc(F)cc1)=CC(C(N1CCC(N(C(CC=CCC)=O)CC)C1)=O)C N1(C(C2(C)CC2)=O)CC2(CC(NC(c3cn(CC(N)=O)nn3)=O)c3nccn32)C1 C(=O)(C(F)CC(CC)CC)NCC1C(CC)CN(C(=O)C(C)=CCO)CC1 c1(C(N2CC(C)N(C(=O)CCC3CCCCO3)CC2)=O)nncc2c1CCCC2 C(C(O)CC(=O)NCCCCc1ncc[nH]1)NC(Cc1n(C)ccc1)=O N1(C(C23CCC(OC)C2C3)=O)CCN(C)CC1C(=O)N(C)Cc1ccnn1C S(=O)(=O)(c1ccc(N(C)CCNC(=O)N(C)C)c(Br)c1)N1CCC(COCC)C1 C(=O)(C(F)C(=O)NCC1(CNC(c2ccccc2C2CC2)=O)CCC1)OCC c1(C(=O)NC(CC)CNC(=O)C(CO)NC(=O)C(F)(F)F)cc2sc(C)cc2s1 N1(C(c2c(CNC(C(CCC)OC)=O)cnn2C)=O)CCC(=O)N(C)CC1 N1(C(C2(NC(CNC(=O)OCC=C)=O)CC2)=O)CCC2(CC1)CC2C#N C(CC(=O)NOC1CCCC1)N(C(=O)CC1CCC1)CCCO c1(CNC(C2COCCN(Cc3cc(O)ccc3Cl)C2)=O)ccc2c(c1)OCCO2 C(=O)(CS(=O)CC(F)(F)F)NCC1(c2ccc(C(C)(C)C)cc2)CCC1 N1(C(C2CC(CC)C2)=O)CCC(NC(=O)Cc2ccc(CO)cc2)C(O)C1 C(=O)(C1=CCSC1)N1C(CCNC(C(C)OCCC(C)C)=O)CCC1 c1(SC)cnn(C)c1C(=O)NCC(O)CN(C(=O)C(C)(C)CO)C C1(NC(c2c(C)csc2)=O)CCN(C(c2cc(N)c(F)cn2)=O)CC1F c1(N(c2cccc(F)c2)CCC(=O)NCC(=O)OC(=O)C=CCl)ccccc1Br C1(C(=O)C2CC2)CCC(NC(C)(C)C(=O)NC)CN1C(=O)OC(C)(C)C.CO N1(C(c2c(C)noc2)=O)CCC2(CC2NC(C2CCCC(=O)N2C)=O)C1 S(=O)(=O)(CC#Cc1ccccc1)NC(C1CC(C)OC1=O)=O C1(NC(Cn2ccc(C)n2)=O)CCC2CN(C(C3(C#N)CC3(C)C)=O)CC2C1 C1(C(NCP(C)(C)=O)=O)CC2CC2N1C(c1ccn(C(F)F)n1)=O N1(C(C2OCCC(C)C2)=O)CCC2(CCCN(C(=O)CCc3cnc(O)[nH]3)C2)C1 CCN=C(NCCCCCC(C)(F)F)NC1CCC(c2cccc(OC)c2)C1 n1(CC(=O)NC2CC(NC(Cc3cc(C)nn3C)=O)C(O)C2)nc(O)ccc1=O Cc1ccc(C)c(NCC(C2CCC2=O)C)n1 C1(NC(CSCC(=O)NCC(CN(C)C(c2ccsc2)=O)O)=O)CCCCO1 CN1CC2CCC1C(CNC(N1CC(c3ccccc3)CC(C)(C)C1)=O)C2 c1(C(N2CC(NC(Cc3ccc(C#N)cc3)=O)C(O)C2)=O)cc2c([nH]1)CCCC2 CC(C)C(C)C(=O)N(CCC(C(C)C)NC(c1ncoc1CCC(F)(F)F)=O)C c1(COC)ccoc1C(=O)NC(C)C(C)NC(c1ncccn1)=O n1(CC)ncn(NC(=O)c2cc(CNC(=O)C(C)(O)C3CCC3)[nH]n2)c1=O Cc1nc(N2CCN(C3CCCN(C(C4CC4C)=O)C3)CC2)c2scc(C)c2n1 C(=O)(C1=CCCOC1)NC(C)CN(C)C(c1cnc(N(C)C)s1)=O N1(C(C(C2CC2)OC)=O)CCOCC1C(=O)NCCN1CCNC1=O CCC(CC)(CC)C(c1ccccc1)N(S(=O)(=O)CC(=O)OC)C C1(NC(CCCOC(C)C)=O)CCN(C(=O)CCC2CC2(C)C)C1C N1(C(C(C)OC(C)C)=O)CCC2(CC1)CC(C(=O)Nc1nccn1C)CCO2 N1(C(c2c(C)ncs2)=O)CCCC(NC(=O)CC2CC3CC3C2)C1C Cc1oc(Cl)nc1C(=O)N(C1CCN(C(=O)CC2CCOC2C)CC1)C1CC1 Cc1cc(C#N)cnc1N1CCC(C)C(NC(C2CC(n3cnnc3)C2)=O)C1 C1(OC)CC(CCNC(=O)CC2CCC(=O)N2)N(C(=O)Cc2nc[nH]n2)C1 C(C)(CNC(=O)CC1CCC(=O)CC1)(CC(C)C)NC(Cn1c(C)cc(C)n1)=O C12(C(=O)NCC3(OC)CCN(C(C4(C#N)CC=CCC4)=O)C3)CCC(CC1F)C2 C1(C(=O)NC(C=C)C)(NC(=O)CC23CCCC2C3)CCCC1C C1(C(=O)NC(C2CN(C(=O)CC(O)C3CC3(Cl)Cl)C2)C)C2CC3C(C2=O)C13 c1(NC(NC2(C#N)CCN(C(C)=O)C2)=S)ccc2sncc2c1 C1(CC(=O)NC2CC(C)(CNC(c3cnc(C)[nH]3)=O)C2)CCCCC1O c1(C(=O)NC(CN(C(c2ccn(CCC)n2)=O)C)C)c(C)[nH]cc([N+](=O)[O-])c1=O C1(CC(=O)NCC2CCC(NC(=O)Cc3ccno3)CC2)CN2CCN1CC2 C(=O)(CC(=O)NCC(C1CC1)NC(=O)Cc1cncn1C)OC N1(C(CC2CCCN(C)C2)=O)CC2CC(NC(c3cncnc3)=O)C(C2)C1 Cc1ncnc(C(=O)NCCC(C)N(C)C(C2CC(=O)NC2(C)C)=O)c1C C(CC(C)(C)C)N(C(C(C)N(C(C1CCCOC1)=O)C1CC1)=O)C1CC1 CC(C)CC(C(=O)N(CC(C)N(C)C)C)ONC(=O)C(C)(O)C1CCC1 C1(CC(=O)NC2CC(N(C(CC=CC(CC)C)=O)C)C2)CCOCC1(C)C C(=O)(N=c1cc(C)o[nH]1)NC(C)C(=O)NCc1cccc(C)c1.C1(=O)C(C)CN1 N1(C(C(CCSC)NC(C2CC(F)(F)CS2)=O)=O)CCn2nc(C)cc2C1 N1(C(c2nc(C)oc2C)=O)CCCC(C2CCN(C(=O)C(C)(C)CO)CC2)C1 CC(C)C(C)C(=O)NCCN(C(=O)CCC1CCC(=O)NC1)CCCN(C)C c1(OCCN(C)C)cncc(C(=O)NC(C)(C)C(O)c2ccccc2)c1 c1(NCC2CC3(CN(Cc4cc(C)nc(C)c4)C3)C2)ncnc2cnn(C)c12 C1(NC(c2cnn(CCF)c2)=O)CN(C(c2cccc(F)c2)=O)CC12CC2 N1(C(c2cc(C)cc(OC)c2O)=O)CCCC2C1CCCN2C(C)=O C(=O)(N=c1cc(NC(C)=O)n(C)[nH]1)C1C2(CCN(C(c3scc(OC)c3)=O)C2)C1 C(=O)(C1CCCCc2ccccc21)N(CCCNC(C(CSC)(C)C)=O)C(C)C C1(CNC(C(C)NC(c2cnc(O)c(F)c2)=O)=O)CC2(CCO1)CC2 c1(C(=O)NCC2CCCN(C(C(CC)C(C)O)=O)CC2)cc2cccnn2c1 c1(OC(CCc2c(OC)nccc2)=O)ccc2c(c1)oc(=O)n2C C1(NC(c2ccnc3ccnn23)=O)CN(C(=O)C(F)OC(F)(F)F)C2(CCC2)C1 Cc1ccc(C(=O)NCCN(C)C)cc1.N12CCCC(C1)n1cc(nn1)C2 C1(NC(CCNC(=O)CO)=O)CC2(CCN(C(C3CCCC(O)C3)=O)CC2)C1 c1(C(=O)NC2CC(C(C(=O)NC(CC)C(C)(F)F)F)C2)c[nH]c2cnccc12 N1(C(C2CC3(CCC3O)C2)=O)CCC2CN(C(C3(C#N)CC=CC3)=O)C2C1.C C(=O)(C(CC)CCOC)NC1(CNC(C(CC)CC)=O)CCCC1 C1(C(=O)NC2C(C#C)CCC2)CC2CC1CC2NC(c1ccn(C(C)C)n1)=O C1(CNC(c2ccc(Cl)nc2)=O)COCCN(C(=O)C=Cc2cccs2)C1 C1(C(=O)OCC2N(C(=O)OC(C)(C)C)CC3(CC3)C2)CCC2(CC1)CC2C#N c1(NC(C2(C)CCN2C(=O)Cn2cc([N+](=O)[O-])cn2)=O)cc(Cl)nnc1Cl C(=O)(C1CCOc2c(F)cccc21)N1CCCCC(NC(C(=O)NC2CC2)=O)C1 N1(C(C2CCN(C)C2)=O)CC2CCCC(NC(=O)CC=C(Cl)Cl)C2C1 N1(CC2N(C)CCCC2)CCC2(CC(CO)C2)C1 C1(CCC)CC(C(=O)N(C)CC2CCCN2C(=O)C(CC)n2cncn2)CCO1 C1(CCNC(CC(CC)C)=O)CCN(C(=O)CC2(CSC)CC2)CC1(F)F C1(C(=O)NC2C(NC(c3ccn(C)c3)=O)COC2)CCOC1(C)C c1(OC)cc(C(=O)N(C2CCCN(C(=O)CN(S(C)(=O)=O)C)C2)C)nn1C C12(C(N3CCC(NC(c4n(CC=C)ccc4)=O)C(C)C3)=O)CC1COC21CCC1 c1(C(=O)NC(CCC)CCc2ccccc2)coc2c1C(=O)NCCC2 c1(CNC(C2CC(n3cc(CC4CC4)nn3)C2)=O)cc[nH]c1C(=O)NC1COC1 C(=O)(C(O)CCCNC(c1ccc(C(N)=O)[nH]1)=O)N(CCOC)C(C)C1CC1 N1(CC)OCC(OC(c2ccnc(Oc3cccnc3)c2)=O)C1=O N1(C(=O)CC2CC2)CCCCC1C1CCCN1C(=O)C(C1CCCCCCC1)O CCS(=O)(=O)c1cccc(C(=O)NC2CC(n3cc(C4CCC4)nn3)C2)c1 C(CC(C(=O)NCCn1cnnc1)NC(=O)C(c1cnn(C)c1)=O)=CC CC1(C)CC1(C(=O)O)NC(=O)Cc1nc(-c2cccs2)n[nH]1 c1(NC(=O)CCc2ccncn2)ccnc2ccnn12 N1(C(CCCCCOC)=O)CC2CCCC(C1)N2C(=O)C1CCCc2cncn21 c1(C(C(=O)NC(C)(CNC(C2CCNC2=O)=O)C2CC2)=O)c[nH]c2ccccc12 C1(C2CCC2)(C(=O)NCC2(C)CCCN(C(C(C3CCC3)OC)=O)C2)CC1(F)F C1(CC)CC(C(N2CCC(OCCNC(=O)COC(C)CC)CC2)=O)CCO1 c1(CC)conc1C(=O)NC(C(=O)NCCc1ncnn1C)C1(O)CCC1 c1(C(=O)NC2CN(C(C3(C#C)CC3)=O)C2)ccc2c(c1)NC(=O)NC2 [N-]=[N+]=NC1(C(N2CCCC2C(N)=O)=O)COC1 c1(CSNS(C)(=O)=O)ccc(-c2ccc(C(=O)NC3OCC(C)C3)s2)cc1.C1CN1 CCCCC(CC)C(=O)NCC1(OC)CN(C(=O)C(C(C)(C)C)NC(=O)OC)C1 C1(CCCC)CCN(C(=O)C(C2CC2)N(C(=O)C=C(C)C2CC2)CC)CC1 C(=O)(C(F)CCC(C)C)N1C(C)(C(=O)Nc2c(C)nn(C)c2)CCC1 C1(n2cc(-c3c(C)cnn3C)nn2)CC(C2CC2)=NO1 c1(OC)ccc(C(=O)NCCNC(C2CCN(C)C(=O)C2)=O)c(Cl)c1 c1(C(=O)NC2CC(F)(CNC(C3CCS3(=O)=O)=O)C2)c[nH]c2cc(F)ccc12 N1(C(C(CCC)C(C)C)=O)CC(C2CCCCN(C(C3CN(C)C(=O)N3)=O)C2)C1 C(C(C)(C)C(C)(F)F)(c1nnnn1-c1ccc(F)cc1)NC(C1CCOCC1)C C1(NC(C(C)NC(c2cccs2)=O)=O)CCC(NC(=O)C(C)(F)F)C1 c1(CC(=O)NC(C(C)NC(c2cc(CC)n(C)n2)=O)C(C)C)c(Cl)cccc1Cl N1(C(C(CCC)NC(N)=O)=O)CC2CCC(C1)N2C(c1cccc(=O)o1)=O N1(C(c2nccc(COC)c2)C(=O)NC2COC2)CCOCC12COC2 CC(C)CC(C)C(=O)N1CCCC(C)(CNC(c2cc(CO)ccc2Cl)=O)C1 CCC(CC(=O)N1CCC2C(C(=O)NCCCC(=O)OC)C2C1)C1CC1 C1(C)(C(N(CCCOCCN(C(C2C(C(=O)OC)CC2)=O)C)C)=O)CCCO1 C1(C(=O)NCC2CN(C(=O)C3=COCC3)CC2(F)F)(OC)CCCCCC1 c1(C(N(C)CCNC(=O)COCCCF)=O)sccc1S(N)(=O)=O C1(NC(C2N(S(CCC)(=O)=O)CCC2)=O)CN(C(=O)CN(C)CC)CC1N=[N+]=[N-] Cc1cnc(N(CC(C)NC(=O)CC2C(C)(C)C2(C)C)C)nc1S(C)(=O)=O C(=O)(C(C)(C)C(C)O)N1CC(OC)C(NC(=O)Cc2ncccc2C)C1 c1(CNC(C(c2ccco2)NC(CCN(CCC)C)=O)=O)ccncc1C C1(C(=O)NC2C(CNC(C(C)OC)=O)CCC2)CC(=O)N(c2ccccc2Cl)C1 CC1CNc2c(C(=O)NCC(C3CC3)NC(=O)COC3(C)CCCC3)cnn2C1 N1(C(CC=CCC)=O)CC2(CCCC2NC(c2ncn(C)c2C)=O)C1 n1(CC)cc(C(=O)C(N2CCC(CNC(=O)CCNc3ccccc3)C2)=O)cn1 N1(C(C2(C(=O)OCC)CC=CC2)=O)CCC(CNC(=O)C(=O)NCC)C12CCC2 N1(C(C2(OCC)CCC2)=O)CCCC(C=O)C1.N1(C2(CC(=O)N)CC2)CCCC1 c1(C(=O)NCc2c(F)cc(C)c(F)c2)c(F)cncc1C1=CCN(C)CC1 C1(CNC(CN(C(C)C)C)=O)CCC2(CN(C(c3cc[nH]n3)=O)C2)O1 C=C=C(C)CC(=O)N1CCC(C2CCCN2C(C2CSCN2C(C)=O)=O)C1 N1(C(c2cc(C(C)C)no2)=O)CCCCC1CN1CCOC1=O Cc1cccnc1CCC(=O)NC1CCCC(C(=O)NC(C)(C)C)C1 CCC(CCC(=O)N1CCN(C(=O)CCSC)C2CC12)OC C1(CNC(Cc2c(C)n(C)cn2)=O)CN(C(c2cscn2)=O)C(C)(C)C1 c1(C(N2CC(CC(=O)NC(C(=O)OC(C)C)C)OCC2)=O)ncc(F)cc1F C(=O)(CC1=CCCCC1)N1CCCCC(CCC(=O)NC2(C)C(C)CCCC2)C1 C1(C(=O)NC(CCC)C(F)(F)F)C(C2CC2)CCN1C(=O)CN1CCNC(=O)C1 C1(C(=O)OC(C)C)(CN(C(=O)Nc2nccs2)C(C)C)CCc2ccccc2O1 c1(C(=O)NCCOCCNC(C(C(=O)OCC)C)=O)c(OC)ccnc1F c1(NC(=O)OC)cccc(S(=O)(=O)N(C)C(c2ccc(NC)cc2)=O)c1 N1(C(C(Cc2ccccc2)OC)=O)CCCC(CNC(c2cc(CF)on2)=O)C1 C1(C(=O)NCC(C(=O)NC)(C)C)CN(C(=O)C(OC)OC)CC12CC2 C12(C(=O)OC)CC(C(=O)NCC3CN(C(=O)CCc4cnccn4)C3)(C1)C2 N1(C(CCNC(N)=O)=O)CCC(CN2CCN(C(C3CC3C(N)=O)=O)CC2)CC1 C(=O)(C(O)CC(C)(C)C)N(CCCCCC(=O)N(C)Cc1nc(=O)o[nH]1)C Cc1cc(C(=O)NC(C2CN(C(c3cc(C)[nH]c3C)=O)C2)C)n(C)n1 CCC(C(=O)NCC(F)CNC(=O)C=CSC)OC1CCCC1 CCCC(C(=O)N1CC(NC(=O)Cc2cc(C3CC3)no2)C1)S(N)(=O)=O N1(C(C2(C)C(C)C2)=O)CC(C2CC2)(C(=O)NCC2CC(C#N)C2)C1 C1(NC(C(CCCCC)F)=O)CCC2(CCCN(C(c3ccc(Cl)o3)=O)C2)C1 CC(COc1ccc(F)cc1)N=c1ccnc(NC2CCCC(C)(C)C2)[nH]1 C#Cc1cccc(C(N2CCCCCCC2)C(=O)NC(C)C)c1 CCC(C(=O)N1CCC(CN(C)C(c2sc(C3CCCC3)nc2C)=O)C1)C(C)C C1(CNC(=O)CCF)COCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(c2ccc(F)cc2)C)=O)CCC(C)C(NC(=O)Cc2ccc(F)cn2)C1 C=CC(C)CCNC(c1occc1CNC(=O)C(c1cnn(C)c1)O)=O N1(C(CN2CC(C)(C)C2)=O)CC2(CCC(CNC(C3CC=CCO3)=O)O2)C1 c1(NC(c2cc(-c3ccc(Cl)c(C(F)(F)F)c3)[nH]n2)=O)ccc2nncn2c1 N1(C(C2C(C3C(C)C3)C2)=O)C2CCC1(CNC(=O)C(C)(C)C(F)F)CC2 c1(-n2cc(CCNC(=O)CCCOCc3ccccc3)nn2)cc(F)ccc1Cl C1(NCc2c(C)nns2)CC(NC(=O)C(=O)NCCC(F)(F)F)C1(C)C CN=c1ccc(C(N2CCCC(C(C)NC(=O)COC(C)C)C2)=O)c[nH]1 C12(C(=O)NCC(CNC(Cn3ncn(C)c3=O)=O)(C)O)CCC(CO)(CC1)CC2 C1(CC(=O)N(C(C)C)CCNC(=O)C(C)(C)c2ccns2)CCCCN1C c1(C(=O)NCC2C(CNC(C3N(CC)CC3)=O)C2)ccc(S(=O)CC#N)cc1 C(=O)(C1=NNC(=O)CC1)NCC1(CNC(c2cccc(NC)n2)=O)CC12CCC2 c1(CNC(C)=O)cccc(C(=O)N(C)CCN(c2ncncc2I)C)c1 CC(C)C(C(=O)Nc1ccccc1)NC(=O)OC(C)C.C1C(O)CNC(=O)N1 c1(CNC(CS(CC)(=O)=O)=O)cc(C(=O)O)c2c(c1)CCO2 C=CC1CCCN(C(c2cnccc2Br)C(=O)N(CC)Cc2nnn(C)n2)C1 N1(C(CC2CC(NC(C3CCC(N(C)C)C3)=O)C2(C)C)=O)CC2(CCCC2)C1 n1(CCC=C)cc(CCC2(O)CN(C(C3(CCS(N)(=O)=O)CCC3)=O)C2)nn1 N1(C(C2CCC(C)(CC)O2)=O)CC(C)N(C(=O)Cc2cnn(C)c2C)C(C)C1 n1(CC)nc(C(=O)Nc2ccc(CN3CCOCC3)c(Br)c2)c2c1CCOC2 C(=O)(CCCC(=O)NC1CC1)N(C)CCN(C(=O)C(F)n1ccnc1)C c1(CC)cc(Cl)ccc1C(=O)OCc1ccnc(C(F)F)c1 C(=O)(CS(C)(=O)=O)N.C(=O)(C(F)C1CCOC1)N(CCCN(C(=O)CO)C)C C1(C(=O)NCCC2(CNC(C(CC)(C)C)=O)CC2)Cc2cccnc2C1 Cc1nc2cccc(C(=O)N(C(C)CCNC(=O)C(c3cccnc3)O)C)n2n1 CCCC(C)C(=O)NCC1CCCN1C(=O)CN(CC(=O)N(C1CC1)CC)C C1(C)(CNC(c2cn(CCC)nn2)=O)CCN(C(=O)CC(=O)N(C)C)CC1 c1(CN(C(C2CCN(C(C3CC3F)=O)C2)=O)Cc2ccc(Cl)s2)ccccc1 CCCC(C)(C)CC(=O)NC1CC(C(N2CC3(CC3)CC2C)=O)C1 C1(CC)CCN(C(=O)COCC(=O)NCCF)C1CC C1(N(C(Cc2ncc(C)s2)=O)C)CN(C(c2ccnc(C(C)(C)C)c2)=O)CC1O C1(CSC)CC(O)CN1C(=O)C(C1(O)CCC1)NC(=O)Cn1[nH]cnc1=N C(=O)(C1=CCN(C)C1)NC(C(=O)NCc1cnc(COC)[nH]1)c1ccco1 CC1=C(C(=O)N2CCCC(NC(=O)C=C3CCN(C)CC3)C(F)C2)CCCO1 CC1CN(C(c2nncn2C)=O)CC1CNC(=O)CCCc1nc(C2CC2)no1 Cc1nn(C2CC2)cc1C(N1CCC(CNC(C2(C(F)(F)F)CCCC2)=O)C1)=O N1(C(C(CNC(CC(COC)(C)C)=O)CC(C)C)=O)CCC2C(=O)NCC2C1 C1(NC(c2[nH]nnc2C2CC2)=O)CN(C(c2ccc(O)nn2)=O)CC1O N1(C(C2C3CN(C)CC32)=O)CCC(NC(=O)Cc2cnc[nH]2)C(F)C1 N1(CC(=O)N(c2cccnc2)C)CCN(C(=O)CO)CC1 C1(C(C(=O)NCC(C)N(C)C(C2CC2(Cl)Cl)=O)C2CC2)CCCCC1 C=CCC(CC(C)C)C(=O)N1CCCC(CC)(NC(=O)C(O)CC2CCCC2)C1 n1(CC)nc(C)cc1C(=O)N(CCC(=O)NCC(c1ccnn1C)O)C c1(OC)noc(C2CC2)c1C(N1CCC(N(C(=O)CCC2CCC2)C)CC1)=O c1(CC(N2C(CCNC(CCC3C(C)C3)=O)CCC2)=O)ccc2c(c1)CCCC2 c1(C(CNC(CC=C=C)=O)NC(c2n[nH]cc2Cl)=O)ccccc1F N1(C(C2C(C)C2)=O)CCCC2(C1)CN(Cc1cc(Cl)ncc1C(F)(F)F)CCO2 C(=O)(C1CC=Cc2ccccc21)NCC(CNC(C1(F)CCCCC1)=O)O c1(NC(C2CC2C(=O)NC2CC(F)(F)C2)=O)cc(C(=O)OC)ccc1OC(C)=O c1(CC)oc(C(N2CC(O)CC2C(N2C(C)CC2(C)C)=O)=O)cc1C C1(CC(=O)NCC2(C(=O)OC)CNC2)(CN(C)C)CCCCC1 C1(C(N2CCN(CCN(C)C(c3c[nH]c(=N)s3)=O)CC2)=O)(OC)CC2CCC1C2 CC(CC(=O)NC1(CF)CCN(C(=O)CN2CCCCC2=O)C1)C(F)(F)F c1(CC)ccsc1C(=O)NC(C)CN(C(=O)CCc1ncc[nH]1)CC C1(CCCNC(C2COC(=O)C2)=O)CN(C(c2sccc2Cl)=O)CCO1 c1(CCCN2C(C)(CO)CCC2)ccc(F)c(F)c1 CC(O)CC(C)N=c1ccnc(NCCC23CCCN2CCC3)[nH]1 N1(C(C2(C)CCCN(C(C3ON=C(C)C3)=O)C2)=O)Cc2ccc(F)cc2C1 N1(C(C(C2CC2)OCC)=O)CCOC2(C1)CN(C(C1CC1C(F)F)=O)C2.C1(C)CC1 N1(C(c2c(CC)ccs2)=O)CCCC(NC(C23CC(C2)C(C)(C)O3)=O)CC1 C12(NC(CC3CC(OCC)C3)=O)CCC(CC1)N(C(=O)CC1(O)CCCOC1)C2 O=C(CC1NC(=O)c2ccccc21)NCCOC1CN(C(C2CCC(=O)N2)=O)C1 C1(C(N(CCC(=O)OC)C)=O)CCN(C(=O)CC2CC(SC)C2)CC1 C#CC1(NC(C2(C(=O)O)CC(c3cn(CCCCF)nn3)C2)=O)CC(F)(F)C1 CC1(C)CC(CNC(c2cnccn2)=O)CN(C(=O)CCCS(N)(=O)=O)C1 Cc1cc(C(=O)N(CC(C)O)CCNC(=O)C(C)(F)F)cc([N+](=O)[O-])c1Cl c1(C(=O)NC(CN(C(=O)CC2CC2(Cl)Cl)CC)C)cc(N)ccc1[N+](=O)[O-] CCN=c1ccc(C(=O)NCC2C3CN(C(=O)CSc4nnnn4C)CC23)c[nH]1 N1(C(C=CC)=O)CCc2c(CNC(=O)CCCN3C(=O)CNC3=O)cccc2C1 c1(OC)ccc(C(C)CNC(=O)NC2CC2c2cn(C)cn2)cc1OC Cc1ccc2c(cnn2C)c1-c1csc(NC(C2CC23CCOC3)=O)n1 CC1(C#N)CN(C(c2sccc2CN=[N+]=[N-])=O)C1 CC(C)CCN=C(NCC1CCOC1(C)C)NC1CCC(=O)NC1 C1(CN=C(NCC(F)F)NC2CCOC(c3cccc(F)c3)C2)CC2(CCCC2)C1 Cc1cccnc1C=CC(=O)Nc1cn(C)nc1C(F)(F)C(F)(F)F C(=O)(C(C(C)NC(C1C(C)(C)C1(C)C)=O)C(C)C)N(C)Cc1cc(OC)no1 c1(CC(=O)NC2C3CN(C(CC4CN(C)C4)=O)CC32)c[nH]c2cc(F)ccc12 c1(C(=O)NCC2N(C(C3C(C(C)C)C3)=O)CCCCC2)cc2cccnc2o1 N1(C(=O)Cc2c[nH]nc2C(F)(F)F)CC=CC(NC(=O)CC2(O)CCOC2)C1 c12ccc3nnc(n3c1)c(=O)[nH]c1ccc2cc1.c1(CC)cc(C(N)=O)n(C)n1 c1(C(N2CC(O)(C(C)NC(=O)C(C)n3cncn3)C2)=O)cc(CO)n(C)n1 C(CO)(CCCCNC(=O)C(F)=C1CCCC1)NC(=O)CCC1CCC(O)CC1 C(CC(C)C)(C(=O)N1CCC(F)C(O)C1)ONC(=O)C1C(=C)C1 c1(C(C)NC(CN(CCOC)C(c2cnn(CC3CC3)c2)=O)=O)ccc(C)cc1 CC(C)CC(O)C(=O)NCC(C1CCC1)NC(=O)CC1(O)CCCN(C)C1 C1(C(N2CCC(OCCNC(c3cc(C)c(C)s3)=O)C2)=O)CCCN2CCCC12 C(=O)(C(O)C1=CCCCC1)N1CCCC(CCC(=O)N(CCOC)CCF)C1 c1(OC)cccc(F)c1CNC(=O)CC1CN(Cc2ncccc2OC)C1 c1(C(=O)NCC2CC(OC)CN2C(C2OCCC2C(C)C)=O)cc2occc2[nH]1 C1(NC(C(C)(C)OC)=O)CN(C(=O)C(C(C)C)c2ccc(Cl)cc2)C(C)(C)C1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)cnn2C)=O)ccccc1CC C(=O)(C#CC(C)(C)C)N(CCCN(C(=O)COC1CC1)C)C CCCCCCC(C)C(=O)NC1CN(C(=O)C=Cc2ccc(C(N)=O)o2)CC1(C)C N1(C(CN(C(COC)=O)C)=O)CCC2CCC12CNC(c1cccc(F)c1N)=O C(=O)(CC(C)(C)CCC)NC(C1(O)CCN(C(C2(CC=C)CCOC2)=O)CC1)C CC(C)CC(O)C(C)C(=O)N1CC2(CCC2)CC1C(=O)NCC1CC2C=CC1O2 N1(C(c2c(SC)cccc2)=O)CC(CNC(=O)C(C#N)C(C)(C)C)C2(CCC2)C1 C1(C)(CC(=O)NCC(c2cnn(C)c2)C)CCN1C(c1cnn(CCF)c1)=O C1(C(=O)NC2CC3(C(C(=O)Nc4ccc(N(C)C)nc4)C3)C2)CC2CC1CC2=O N1(C(CCC2N(C(c3c(C)cc[nH]3)=O)CCCC2)=O)CCOCC(O)C1 C1(OC)CN(C(C23CCCC2C3)=O)CC1NC(c1ccccc1C1CC1)=O Cc1cc(CN=c2[nH]c(C(=O)NCCCN3CCCC3)cs2)cc(Br)c1 CC1(C)CC(NC(c2c(F)cccc2Cl)=O)CN1C(=O)CC1CC1 Cc1cc(N(C(=O)C(C)(C)C(C)C)C)c(O)cc1F N1(C(C(C(C)(C)O)F)=O)Cc2n[nH]cc2C1C(=O)N1CC(OCC23CC(C2)C3)C1 c1(N(C)C)nc(Cl)c(C(N2CCOCC2CNC(=O)CCc2cnc(O)[nH]2)=O)s1 C=CCC(C)(C)CC(=O)NCC(C)CN(C)C(C12COC(CO)(C1)C2)=O N1(C(C(=O)NCN(C)C)=O)CCCC(NC(=O)CN(c2ccncc2)C)C1 CC1CC(NC(=O)C(F)(F)c2nccn2C)CCN1C(=O)CCC1CC1(Cl)Cl C1(CNC(CSCC(C)C)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1(F)F c1(OC(C)C)ccccc1C(N1CCC(OC(c2scnc2Cl)C)C1)=O C1(C(=O)NC(C(Cc2cc[nH]n2)SCC=C)=O)(CC)CN(C(=O)C=CCF)C1 CC1(C)C=C(C(=O)NC2CCN(C(=O)CCCCCc3cccs3)C23CC3)C1 C=CC1CCCN(C(=O)CC2CCCCN2C(c2sc(O)nc2C)=O)C1 C12(C(=O)NCC3(CN(C(c4c(C)c(Cl)ccn4)=O)C)CC3)CCCN1CC(O)C2 C1(CC)CN(C(c2cnc(C(F)F)c(C)c2)=O)CCN1C(=O)C(O)CN(C)C C1(C(N)=O)COCCN1C(C12CC1CN(Cc1ncccc1F)C2)=O C1(CNC(C=C(C)C(F)F)=O)CCC(N(C(=O)CC2COCCO2)C)CC1 c1(C(N2CCC(C)(CNC(=O)C(F)C3CCC3)C2)=O)cc2ccccc2s1 c1(CNC(C2C(Nc3ncc(C(N)=O)cc3Cl)C2)=O)cn2cc(F)ccc2n1 CCCCC(O)C(C)C(=O)NC1CC(CC(N2CCC2(C)C(=O)NC)=O)C1 c1(CNC(=O)CC(C)(C)CNC(C2C(c3n(C)cnc3)C2)=O)cnn2c1OCC2 C(c1c(Cl)cccc1Cl)=CC(=O)NCC(C)N(C(=O)CCc1cnccn1)C C1(C(=O)NCC2C(NC(c3cccc4c3COC4)=O)C2)CCc2ccccc2C1 c1(C(N(C)CC2CN(C(c3scc(OC)c3)=O)C2)=O)ccc(F)c(N(C)C)c1 c1(NC(c2ccc(OCC(F)Cl)cc2)=O)cccc2ncnn12 N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(C2CC2N2CCOCC2)=O)C(C)(C)C1 N1(C(C2C(C(=O)OCC)CC2)=O)C(C(N2CCC(O)(C(C)C)C2)=O)CCC12CC2 c1(NC(CC(c2cn(C)nc2)NC(=O)C=CC(F)(F)F)=O)cccc(C#N)c1 c1(CNC(c2c(C)nc(Br)s2)c2nnnn2C(C)C)cccc2ncccc12 c1(C(N(CCCN(C(CC2C(C)C2)=O)C)C)=O)cn2c(n1)COCC2 N12CCOCC(C1)NC2=O.c1(NC(C2CC=C(C)CC2)=O)ccc(C)c(O)c1 C1(C)(C(=O)NCCCCC(C)NC(C(C)CCO)=O)CCN(C)C1=O c1(C(=O)NC23CC(NC(CN4CC(C)(OC)C4)=O)(C2)C3)ncn(C)c1C c1(C(=O)NCC2CC2NC(C2CCc3nncn3C2)=O)ccc2c(c1)CCCC2 C1(CNC(C(CC(=O)OC)C)=O)CC2CCC1N(C(C1COCC(C)O1)=O)C2 Cc1[nH]c2ccccc2c1C(=O)NC1CCCC1(C)NC(=O)CNC=O C1(CNC(C=CC=CC)=O)CN(C(c2cncc(NCC)c2)=O)CC2(CCC2)O1 c1(C(=O)NCC2C(NC(C3(CC(C)C)CC3)=O)CCCC2)ccc2c(c1)C(=O)OC2 C1(C(=O)NCc2c(CC)nccn2)CCCC(NC(=O)C(C)OCC2CC2)CC1 c1(OCc2n(C)cnn2)c(Cc2cn(-c3ncccn3)nn2)nn2c1CCC2 c1(C(N2CCCC(C(C)(O)CNC(=O)C(N)=O)C2)=O)cc2ccc(F)cc2o1 C1(NC(C(C=C=C)C)=O)CN(C(c2cccnc2SC(F)F)=O)CC12CC2 c1(C2(C(=O)NCC3C(CNC(C4CCCC4)=O)C3)CC2)ccc(F)cc1 C1(CNC(CCC=C)=O)CC(C)N(C(c2cn(C(C)C)cc2C)=O)C1 C1(NC(=O)CC2CCC3C2C3(F)F)CC2(C1)CN(CC=Cc1cncc(O)c1)C2 CN1CCC(CC(N2CCC(C(C)(C)NC(C3CC3F)=O)C2)=O)C1 c1(C(=O)NCCOCCNC(C(CC)(C)CO)=O)n[nH]c2ccc(C)cc12 N1(C(C(C)CCO)=O)CCC2(CCCC2CNC(c2cccn(O)c2=O)=O)CC1 C(=O)(CC(O)C(C)(C)C)N1CCC(COC)(NC(C2OCCN(C)C2=O)=O)C1 Cc1nnc(N2CC3CC(NC(C4CCN(C)CC4)=O)C3C2)c(C#N)c1C c1(C(C(=O)OC)NCc2cncs2)ccc(F)c2c1CCC2.CC(C)(C)O C1(C(=O)NC(C)CCCNC(=O)COCC(C)(C)C)CC2(C1)NC(=O)NC2=O CCCCCCC(F)C(=O)N(C1CC(NC(=O)Cc2nonc2C)C1)C C(c1c(F)cccc1F)=CC(=O)NC1CC2CC1N(C(c1ccoc1Br)=O)C2 C1(CC(=O)NC(CCC)CO)CCCN(C(=O)C(N2CCOCC2)C)C1 O=C(CC1CCC2(CCC2)O1)NNC(=O)c1cc(C(F)(F)F)cnc1N O=C(CCC(F)(F)F)NC(C1(O)CCCCC1)C(=O)NC1CC(F)C1 Cc1cc(Br)cc(CN2CCC(N(C)C(c3cnc(O)cc3O)=O)C2)c1O C1(CCNC(=O)OC(C)(C)C)CC(n2c(C)c(C(=O)N)cn2)C12CCC2.C(F)F C1(C(=O)NCC(C)N(C(=O)CCc2n[nH]c(=N)s2)C)CCN(C)C(=O)C1 C1(CNC(C2N(S(C)(=O)=O)CCC2)=O)CCCCCN1C(=O)C1=CCCOC1 c1(OCC)ccc(C(N2CC(OC)C(NC(c3ncsc3C3CC3)=O)C2)=O)cn1 N1(C(C2C(C)(Br)C2)=O)CC2(C1)C(NC(=O)Cc1cccc(F)c1)CCS2(=O)=O N#Cc1cncc(NC(C2CN(C(c3cncs3)=O)CCO2)=O)n1 C1(C(=O)NCCc2nccc(O)n2)(OC)CCN(C(c2ccn(C(F)F)n2)=O)C1 c1(CC)nn(C)cc1CNC(c1c(C)noc1C)c1ccccc1 C=CC1(C(=O)NC2(C)CN(C(C)=O)C2)CCN(C(C23CCC(C2)C3(C)C)=O)CC1 c1(CN(C(C2COCC(C)O2)=O)C)nnc2n1CCNC2=O c1(C(=O)NC2CCN(C(C3(C)CC=CC3)=O)C2)ccc(-c2cc(O)ns2)cc1 c1(CN2C(C(N3CCC(NC(C)=O)C3)=O)CC2)cc(F)cc(Cl)c1 c1(C(N2CC(SC)C(NC(=O)CC3(C)CCCCC3)C2)=O)cc(C)c(C)nc1C c1(C(=O)NC2CC(C)N(C(c3ccn(O)c(=O)c3)=O)CC2)cnn2ncccc12 C1(C(=O)NC2C(NC(C3(CCOC)CC3)=O)C2)CCC2(CCOCC2)C1 Cc1ccc(C(=O)NC(C)CN(C(=O)CCC(=O)c2cccnc2)C)cc1CO C1(C(N2CCC(Nc3ncnc(O)c3Br)C2)=O)CC2(C1)CS(=O)(=O)C2 Cc1scc(C(N2CCC(C)(NC(=O)C=Cc3nnn(C)n3)C2)=O)c1C C12(NC(COCC(C)C)=O)CC(CNC(=O)COCC(c3ccccc3)C)(C1)C2 C(=O)(CCCN(C)N=O)NCCCN(C(c1cnn(C)c1)=O)CC N1(C(CC(=C=C)C)=O)CC(NC(c2cn(C3CC3)cn2)=O)CC12CCOCC2 Cc1ccc(CC(=O)NCC2CCN(C(=O)CSc3nncs3)C2)cn1 C1(CCN(C)CCSCCO)CCN(C(C2CC(F)C2)=O)CC1 Cc1ccc(C=CC(=O)NC2CCCC2NC(c2ncoc2C)=O)cc1C c1(C(N2C(C)CC(CNC(CCSC)=O)C2)=O)coc2c1COC2 C1(C(N2C(C)(CNC(c3scc(C(C)=O)c3)=O)CCC2)=O)CC2(CCCC2)C1 c1(NC(C2CC(NC(CNS(C)(=O)=O)=O)C2)=O)ccc(S(=O)(=O)N2CCCC2)cc1 N1(C(c2c(C)cncc2)=O)CCC2CCC(C1)N2C(=O)CN1CC2CC2C1 CCCC(C)(CCC)C(=O)N1CCOC(CC(N2CC(CC)C(O)C2)=O)C1 c1(CNC(C(c2ccccc2)OC(C)C)=O)nc(C2CC2)sc1Br c1(C(=O)NC(C(C)NC(CC(n2ccc(C)n2)C)=O)C)ccc2c(c1)OCCO2 c1(C(N2CC(NC(C3CCCO3)=O)CC(C)(C)C2)=O)ccc2c(O)n[nH]c2c1 C1(CCNC(C(C)OCC(C)C)=O)CN(C(C2(N(C)C)CC2)=O)CCS1(=O)=O C=CCC(C)(C)CC(=O)NC1CCN(C(c2ccc(CC3CC3)cc2)=O)CC1F Cc1ccc(NC(=O)CC2CCCNC2)nc1SCc1ccccc1 c1(OC)ccc(CN2CCC(NC(=O)C(c3ccc(OC)cc3)C)C2C)cc1O c1(C(=O)NCC#CC(=O)NC(C)Cc2ccnn2C)ccc2cccnn12 c1(C(N2CC3(N(C(C(C)=O)=O)CC3)C2)=O)cc(Cl)c(Cl)cc1I CCC(CC)(CN=c1cc(C(F)F)nc[nH]1)NC(=O)CCOCC1CCOCC1 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(c2ccc(C)cc2O)=O)C2(CCC2)C1 c1(NC(C2CC(NC(C3CCCO3)=O)C2)=O)cc2ccccc2c(Br)n1 Cc1cc(CC(N2CCN(C(c3c(C)coc3C3CC3)=O)CC2C)=O)c(O)c(C)c1 C(=O)(C1=CC2(CN(C(C3CCC(F)C3)=O)C2)OC1)NCCc1n(C)cnc1 C(=O)(CC(C)CC(C)C)NCCC1N(C(CCCc2nnc(C)n2C)=O)CCC1 N1(Cc2cccc(OCC)c2)CC2OCCN(C(C3CCC(F)(F)C3)=O)C2C1 c1(SCC(=O)NC2(CNC(C(c3cnn(C)c3)OC)=O)CC2)ccc(Br)cc1 C1(NC(c2c(N)non2)=O)CC2CCC(C1)N2C(C12CC(c3ccccc3)C1C2)=O N1(C(c2c(C)sc(O)n2)=O)CCCN(C(c2cc(N)cc(O)c2)=O)CC1 N1(C(C(C)c2cc[nH]n2)=O)CCOCC1C1CCCO1 N1(C(CN(C)C(N)=O)=O)CCC(NC(=O)CC(=O)NCC2CC2)C1(C)C c1(C(=O)NCCN(C(C2CC2c2ccccc2)=O)CC)cc(C(C)C)nn1C CC1=C(C(=O)NC2CCN(C(=O)Cc3ccc(F)cn3)C(C)C2)CCS1(=O)=O CC1(C)CCCCC1CC(N1CCSCC1CCNC(=O)CC1CCCCC1)=O c1(NC(C2OCCN(C(c3ccc(C)nc3)=O)C2)=O)c(F)cc(Br)cc1Br C(=O)(C1CC(=O)Nc2cc(F)ccc21)NC1(C)CN(C(C2COC(=O)N2C)=O)C1 c1(OC(C)(C)C)cncc(C(=O)NCC2(C)CCN(C(C34CC(CO3)C4)=O)C2)c1 c1(C(=O)NCCCCCN(C(COC(CC)C)=O)C)cncc(CO)c1 O=C(CC(C(F)(F)F)N1CCOCC1)OCc1cc2ncccc2[nH]1 c1(CCC(=O)NCC2(O)CCN(C(c3cc(F)cs3)=O)C2)ccccc1Cl C12(CNC(C3(NC(CC4CC(SC)C4)=O)CCCC3)=O)CC=CC(C1)OC2 CC1(C)CCCC(C(=O)NCc2ccc(C(N3CC(F)(C#N)C3)=O)o2)C1 C1(NC(CCCNC(C)=O)=O)CN(C(c2scnc2C)=O)CC1C Cc1cc(C(N2CCC(C(C)NC(=O)COCC3CC3)C2)=O)ccc1O C(=O)(C(O)C(C)(C)CC)NCC1CN(C(C(CC=C)(F)F)=O)CC1(C)C N1(C(C(C)NC(=O)C2CC2)=O)CC(CC(=O)NCC2(F)CN(C)C2)C2(CC2)C1 c1(C(=O)NCC(C)NC(c2[nH]cc(C)c2)=O)cccc(C#N)c1Br C1(C(=O)OCC)CN(C(=O)NC2CCCC(O)C2O)CC1(C)C c1(C(N2CC(COC)(CNC(=O)C(CO)N(C)C)C2)=O)cc2n(n1)CCCO2 CC1(C(=O)NC2CC(NC(C3(c4cccnc4)CC(F)(F)C3)=O)C2)COC(=O)C1 CCC(CC(=O)NC(c1n[nH]c(CC)n1)C)OC.C12CC(O)C1NC2=O C=CCC(CNC(c1cc(C(=O)OC)ccc1Cl)=O)C(=O)O Cc1sc(C(=O)NC2(C3CCCN3C(c3cc(O)n(C)n3)=O)CC2)nc1O N#Cc1cccc(NC(C2C3CN(Cc4cccc5ccoc45)CC23)=O)c1[N+](=O)[O-] CCCC(C)CCN=c1ccnc(NCCOc2ccccc2C)[nH]1 N1(C(C(CN(C(c2c(CC)cncc2)=O)C2CC2)C)=O)CCC2(CC1)CC2 Cc1cc(CC2CC(CCc3ccccc3)=NO2)c(Br)cc1F C12(C(=O)NC(C(=O)OCCC)C)CC(C)(CN1C(=O)C(C)S(N)(=O)=O)C2 C1(NC(C(c2scc(C)n2)C)=O)CN(C(C2CC3CCC2CC3)=O)CC12CCC2 c1(C(C)C)cc(C(N2CCN(C(=O)C(F)C(C)(C)O)CC2C)=O)cc(F)c1 O(NC(=O)C(C)N(C)C(c1cccn1C)=O)C(CC)C C1(NC(N(CC)CC2CC2)=O)COCC1O CCCC(CNC(c1ccnc(C)n1)=O)C(=O)N(C)CC1(OCC)CCC1 Nc1cc(C(=O)NC2CCCC(NC(c3cc(F)c[nH]3)=O)C2)cc(F)c1 C(=O)(C1CCCc2sccc21)NC(C(C)NC(Cc1c(C)non1)=O)C(C)C C=C(C)CCC(=O)N1CCN(CC2CCCN(C(C3CC3C(C)C)=O)C2)CC1 N1(C(C=C(CNC(C(COC)N(C)C)=O)C)=O)CC2(CCC(=O)O2)C1 CC(C)P(=O)(CC(=O)NCC1CN(C(=O)CC2CCCC2(F)F)C1)C(C)C N1(C(c2c(OC)c(=O)cco2)=O)CCC2(C1)CN(C(=O)CC(C)CF)C2 N1(C(C(C)C2CCC2)=O)CCC(C(O)CNC(=O)C(c2cccc(O)c2)C)CC1 c1(NC(C2CCN(C(C(COC)OC)=O)C2(C)C)=O)cccc2cccnc12 C=C1CON(C(=O)COC2CN(C(=O)C(CC)N(C)C)C2)C1 C1(C(C(=O)NCCN(C(=O)CC2CCCC2C)CC)F)CCCCC1 C1(NC(C2CC23CCC3)=O)(CO)CCCN(C(c2cnn(C3CCC3)c2)=O)C1 C1(C(=O)OC)CN(C(=O)Nc2cc(C)ccc2Br)CCC1(F)F c1(C(=O)NCC2(C(N)=O)CN(C(c3cnsn3)=O)C2)ccc2c(c1)C(=O)NC2 N1(C(C(CSC)C)=O)CCCC2(C1)CN(C(C1(C#N)CCCOC1)=O)C2 c1(N(CCCNC(c2ccc(CC)o2)=O)C)nc2c(F)cccc2o1 CC(C)C(C#N)C(=O)NCC1CN(C(=O)CCCNC(=O)C2CC2)CC1C c1(OCC)ccc(CCN(C(=O)C(=O)NC(C)(C)C(C)O)CC)cc1 Cc1ncc(C(=O)N(CCCNC(c2ccc(=O)n(C)n2)=O)CCO)c(=N)[nH]1 N1(CCOCCNC(C)=O)CCN(C)CC1.C12CCCN1CC(=O)NC2C Cc1cc(O)c(Cl)cc1C(N1CCC(NC(c2ccc(F)cc2F)=O)C12CC2)=O CCC(C)(C(=O)Nc1ccc(NC(C2CC3(CCCC3)CO2)=O)c(C)c1)C(F)F c1(C(N2CC(O)(C(C)NC(C(C)C3CCCC3)=O)C2)=O)ccc([N+](=O)[O-])cn1 Cn1cncc1C(=O)NC1(CO)CN(C(C2(O)COC2)=O)C1 c1(C(C)C)cc(-c2csc(Cc3ncc(-c4ccccc4)[nH]3)n2)n(C)n1 C12(C(N(CCCC(C)(C)C)C)=O)COC(C1)C(NC(=O)CCC(=O)C1CCCO1)C2 CCCCCC(O)C(=O)NC1CC(NC(C2(CCF)CCC2)=O)C1 Cc1cn2ccnc(C(=O)NCCC(C)N(C(=O)CN3CCC3C)C)c2n1 C(CC(=O)NCC1COCCOC12CCC2)(C(C)(C)C)NC(=O)OC(C)(C)C N1(C(C2N(CC)CC2)=O)Cc2ccccc2C1CNC(=O)CN1CCOCC1 c1(C(N2CCN(CCCNC(C(CCC)OC)=O)CC2)=O)cc(Cl)c(Cl)cc1N N1(C(C(CC)O)=O)CCC(NC(=O)C(C)Cn2cccn2)C(O)C1 C(=O)(CC(C(F)(F)F)NC(C1CCOC1(C)C)=O)N1CCC(CCCC)C1 C1(NC(c2c(F)ncc(OC)c2)=O)CCCC12CN(C(=O)CCCSC)C2 c1(C(N2CC(CC(=O)Nc3ccc(F)c(F)c3O)C2)=O)cc2cccc(Cl)c2s1 O=C(C1=CCCOC1)NCCCNC(c1snc(Cl)c1Cl)=O C1(C(=O)NCC2CC2)C2CC3C(C2NC(=O)COC2(CC)CCOC2)C13 c1(OC)cc(NC(C2CCC3(CCC3)C2)=O)c(C)cc1C c1(C(N2C(c3cccc(OC)c3)CCC2)C(=O)NC(C)(C)C)ccc(C#N)cc1 N1(C(N)=O)CCCC1C(=O)NC1CC(CNC(=O)C(c2ccccc2)O)C1 CC1OCCCC1C(=O)NCC1C2CC1N(C(c1cnccn1)=O)C2 N1(C(C(C)(C)C)=O)CCOC(C(=O)NCC2CC3C=CC2C3)C1 C12(C(=O)NCCCCC3CN(C(C4CC(C)OC4)=O)C3)CCC(O)(CC1)CC2 c1(CC)ccc(C(=O)N(C)CCNC(=O)CCc2cc(C)on2)s1 N1(C(C2(COC)CC2)=O)CCCC2(CCN(C(=O)C#CC3CCCOC3)C2)C1 c1(C(=O)NCCN(C(=O)C(C)C(F)(F)F)CC(C)O)cc(O)nc(O)n1 CCCCCCCCOC(N1CC2CC2(CNC(=O)CCc2ccoc2)C1)=O c1(C(C(=O)NCCCOCC)N(C(C)CC)CC)cc(C)cc2c1CCC2 N1(C(C2CCN2C(c2cc(C3CC3)on2)=O)=O)Cc2ccncc2C1 c1(-c2ccc(C(=O)NCC(CNC(c3c(CC)scn3)=O)O)s2)ccc(Cl)cc1 C(=O)(CS(=O)(=O)C(C)C)NCC12OCC(NC(C(CCOC)C)=O)C(C1)C2 c1(CC(N2C(CNC(CC(C)C)=O)COCC2)=O)ccc2c[nH]nc2c1 CS(=O)CCC(O)C(=O)NCC1CN(C(=O)CC2CC2)C1 c1(C(N(C)CC2OCCN(C(C(CCC)O)=O)C2)=O)nn(C)c(=O)cc1C CN1N=C(CC(=O)NC(c2ccnn2C)C(=O)NCC2(C)CCOCC2)CC1=O C(=O)(C#CC1(C(F)(F)F)CC1)NC(CNC(c1n(C)nc(C2CCC2)c1)=O)CO C1(C(=O)OCC)CCC(NCC2(CC(N)=O)CCCCC2)CC1 Cc1ccc2c(c1)CN(C(C1CCC(NC(C3(C#N)CC3)=O)C1)=O)C2 C1(CC)CN(C(c2csc(O)n2)=O)CCC1NC(=O)Cc1ccc(F)cc1C N1(C(C=C(C)C)=O)CCC(N(C(=O)Cc2ccccc2CC(N)=O)CCO)CC1 c1(-c2cn(CC#N)nc2)c(F)cccc1Br C1(CNC(CC2C(CC)C2)=O)(N(C(=O)CCCc2cnn[nH]2)C2CC2)CCCC1 c1(C(N2CC3(CCC(OC)CC3)C2)=O)cc(C(F)(F)F)ccc1P(C)(C)=O C(=O)(C(C)S(=O)(=O)Cc1ccc(N2CCOCC2)cc1)NCC c1(C(=O)NCCN(C(=O)C(C)(C)F)CC)cc(-c2ccccc2)oc1C CC1(C)C2CCC(C2)C1C(=O)NC1CN(C(C2(F)CC2)=O)CC12CC2 c1(C(=O)NC2CC(C)(NC(=O)Cn3cc(CO)nn3)C2)c(F)cc(Cl)cc1F C(=O)(C(C)S(C)(=O)=O)NC(CNC(C(CC=C)C)=O)(C)C C(=O)(C(CC(=C)C)NC(=O)CC(C)COC)N1CCCC(CCC#C)C1 C1(C(C)NC(c2ccnc(N(C)C)c2)=O)CCN(C(=O)C=CCO)CC1 Cc1cncc(C)c1C(=O)NC(CCN(C(=O)C(C)N(C)C)C)C(C)C N1(C(c2scc(C)c2)=O)CCCC1C1CCCN1C(=O)COCCF c1(C(N2CC(NC(c3cc(OC)ncc3Cl)=O)C(C)C2)=O)nn(C)c(=O)cc1C C1(NC(CCC=C)=O)CCC(C(=O)Nc2cnc(C(C)C)nc2)CC1 C12(C(N3CC(CNC(=O)NCc4c(N)cccc4F)C3)=O)CCCCC1C2(F)F c1(CCNC(=O)NC(C2COC2)C)cccs1.C12CC1C2 C(=O)(C1Cc2ccc(Cl)cc21)N1CC2C(NC(=O)CC3CC3)(C2)C1 c1(NC(N(C(CC)C)C)=O)cnn(CCOC)c1 C1(C)(CNC(c2cccc(CC)n2)=O)CN(C(=O)CCc2ncc(C)[nH]2)CC1C Cn1ncc(C(=O)NC2CCC2NC(=O)C(O)C2CC2)c1Br N1(C(C(COC)(C)C)=O)C2CCC1(CNC(C1CCC(=O)NC1)=O)CC2 N1(C(C2CC=C(C)CC2)=O)CCCN(C(=O)CCNC(C2CCC2)=O)C(CO)C1 Cc1nnc(O)c(C(=O)NCC2(NC(=O)C(C)SC(F)(F)F)CC2)c1C c1(C(=O)NC2C(NC(c3cc(OC)nn3C)=O)COCC2)cccc2nccn12 C1(C(=O)NCCCCC(=O)N2C(C(=O)OC)CCC2)CC2(CCC2O)C1 C1(CC=C)(CNC(=O)C(=O)Nc2ccnn2CC2CCOC2)CCOCC1 C1(OC)CCC(N=c2ccnc(NCc3ncoc3C)[nH]2)CC1 CCC(C#N)C(=O)NC1(CCCCNC(=O)C=Cc2cnccn2)CC1 C1(C(N(C)C)=O)C2CN(C(C3(N)CCC4CC34)=O)CC12 c1(C(N2CC(COC)(NC(=O)C(C)=O)C2)=O)ccccc1OC c1(C(=O)NC2(C)CC(NC(c3cncc(C)c3C)=O)C2)nc2n(c1Cl)CCCC2 C(=O)(C1CCCc2nc[nH]c21)NCC(CNC(=O)CC(c1cccc(F)c1)O)O N1(C(c2cccc(N(C)C)n2)=O)CC(NC(C2(CCF)CCC2)=O)C(C2CC2)C1 C1(C(=O)NC(C(C2CC2)OC)C)CCC=CC1NC(=O)Cn1cnnc1 N1(C(C2C(OC)C2)=O)CCCN(C(C2CC3C=CC2C3)=O)CC1 N1(C(C(CC2CC2)OCC)=O)CCCCC(NC(c2ccc(COC)o2)=O)C1 C1(CN(C(=O)C(O)c2cnc[nH]2)Cc2cnns2)CCOC1=O CC1CCN(C(=O)C(F)OC(F)(F)F)C1C(=O)NCCc1ccoc1 C(=O)(C1CCCc2sccc21)N1CC(C)(NC(c2onc(C)n2)=O)C1 CC1CC(CO)CN(C(C2CCCN(C(=O)CCc3ccnn3C)C2)=O)C1 C(=O)(CC(O)CC(C)C)Nc1ccc(C(=O)NC(CCC)C(F)(F)F)cn1 Cc1cc(C(=O)NC2CCCCC2NC(c2cn(C3CCOC3)nn2)=O)nn1C C(=O)(C(O)C1=CCCCC1)NC(CC)CCC(=O)NCCN1CCC(OC)C1 C1(NC(c2cnn(CC)c2Cl)=O)CC2CN(C(=O)CC3CCN(C)CC3)CC2C1 N1(C(c2cncn2C)C(=O)NC)CCN(C(=O)C=C(C)Cl)CC1 Cc1ccc(CCC(=O)NC2CCN(C(=O)C=C3CC3)CC2C)cc1C C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(C1CCCN1C)=O C1(C(=O)NC(c2cnc(C(F)F)o2)C)=CS(C(F)(F)F)=N1 c1(C(=O)NC2CC(NC(C(C)NC(c3ccc(F)cc3)=O)=O)C2)cn2ccnc2s1 C(=O)(N1CCC(C(=O)NCCC(C)(O)COC)O1)c1c(CC)n[nH]c1 N1(C(c2c(N)non2)=O)CCC(C2CCN(C(=O)C(=O)NCC(F)F)C2)C1 C(=O)(CC(C)C(C)C(C)C)NC(c1cc(C)cc(C)c1)(CC(=O)OCC)C c1(C(=O)NCC(C)CN(C(=O)CCC(F)(F)F)C)cc2c(s1)CCS(=O)(=O)C2 N1(C(CNC(C(C)(C)C)=O)=O)CCC(C)(CNC(=O)CC23COC(CF)(C2)C3)C1 Cc1oc(CO)cc1C(N1CCC(C(C)C(=O)NCCC2CCOC2)C1)=O C(=O)(CCC(=O)NC(C(C)NC(=O)C(=Cc1cccs1)C)C(C)C)N(CC)CC Cc1noc(C(=O)NCC2CC(O)CN2C(=O)CC2CCCC2C)c1C S(=O)(=O)(C=Cc1ccccc1)NC1CCC(NC(c2ccsc2)=O)C1 N1(C(c2c(C)coc2)=O)CC2(CCC2)CC1CNC(c1ccc(CCO)cc1)=O N1(CC#C)CCC(C(N2CC=CC2CNC(C2CC2CC(C)C)=O)=O)CC1 CC(CC(=O)N(c1ccccc1)C1CCCC1)NC(=O)NCCC(N)=O N1(C(C(CC)(C)CO)=O)CCCC2(CCN(C(=O)CC(C)(O)C(F)(F)F)CC2)C1 C(=O)(CC(CN(C)C)C(F)F)N1C(CNC(COCC(C)C)=O)CCC1 C(CC(CC)C(=O)N1CC=CCC1C(=O)NCC1CCC(C)C1)=CC C(C(=O)NC(CNC(c1cccc(SC)c1)=O)C1CCC1)(C(C)(C)C)OC N1(C(=O)C2=C(Cl)CC2)CCCC(C2CN(C(=O)COCCO)C2)C1 c1(CC(=O)NCCN(C(c2cnc(C3CC3)[nH]2)=O)C2CC2)ccc(F)cc1 N1(CCC(N2CC(O)CC(NC(=O)CO)C2)=O)C(=O)c2ccccc2C1=O C1(CC)CCN(C(c2cnn(C)c2COC)=O)C1C(=O)NCCc1cn(C)nn1 N1(C(CCC#C)=O)CCC2CCN(C(=O)CCCCCCCC3CC3)CC2C1 C1(NC(C(C)NC(N)=O)=O)C2CC3CN(C(c4cc5occc5s4)=O)C1C3C2 CC1CN(C(C2(CNC(C3CC(O)C3)=O)CC3(CC3)C2)=O)CC(CO)O1 c1(CC)cc(C(N2CC(CNC(=O)C(c3ccc(Cl)s3)C)CC2C)=O)n(C)n1 c1(C(=O)NCCCN(C)C(C2(CF)CCC2)=O)cncc(C(F)F)c1 C(CC(F)F)(C(=O)NC(C)CN1CCOCC1)N(C(Cc1c(C)nccc1)=O)C C(C)(c1ccccc1C)=CC(N1CC(OCC)(CNC(c2c[nH]cc2Br)=O)C1)=O N1(C(COCC(=O)OC)=O)CCN(C2CCN(C(=O)CCCN(C)C)CC2)CC1 c1(C(N2CC(CC(C)NC(C(CC)(C)F)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl C1(C(N2CCCC(CCNC(C(C)=C(C)C)=O)CC2)=O)CC2CSCC(C1)C2 C(Cc1cc[nH]n1)(C(=O)NCC1COCC1O)NC(CN(C)C1CC1)=O C=CCN=C(NCC1(C)CCN(C(=O)OC(C)(C)C)C1)NC1CC1N(C)C c1(C(N2CCC(NC(c3cnc(OC)c(Cl)c3)=O)C2)=O)c(Cl)cccc1[N+](=O)[O-] C1(CC(=O)NCCC2CCC2)CC2(C1)CN(C(=O)COC1CCCC1)C2 N1(C(C(C)=O)=O)CCC2(CCCCC2N(C(=O)CCc2cc(C)no2)CCC#N)C1 C(CCCCCN=[N+]=[N-])NC(Cn1cc(CNC(C(C)(C)C)=O)nn1)=O C1(O)(C(C)NC(=O)CCc2cn[nH]c2)CCN(C(=O)C(N2CCC(O)CC2)C)C1 CCC(O)C(C)(C)C(=O)N1CCC(N(C(c2sc(C(C)C)nc2C)=O)CC)CC1 C1(=O)N=C2C=C(C)N(N2)N1.CCC(CC)C(c1ccccc1)c1ccccc1 C(=O)(C1=NOC(C(=O)NCc2cnoc2)C1)NC(COC(C)(C)C)(C)C c1(COC(C)=O)ccccc1CC(=O)NC(C)C(C)NC(=O)C=C1CCSCC1 C1(OC)CCN(C(C2C=CCCN2C(=O)CC2(O)CCCC2)=O)C1(C)C O=C1CCC2CN(N3CCOC(c4ccc(F)c(F)c4)C3)CCN12 N1(C(=O)NC(c2cc(C(F)F)co2)C2CC2)CCCC(n2cccn2)CC1 CCC(CC(=O)NC1CC(CNC(c2sccc2-n2ccnn2)=O)C1)C1CC1 C12(C(N3CC(C)C(O)CC3)=O)CCCC1CCN2C(=O)CCOCC1CC1 CC1N(C(=O)NCC2(c3ccccc3)CCCO2)CCCC12CCC2 CC12CC(NC(=O)CCC3CCCCC3)(C1)C1(CN(C(c3ccc(F)s3)=O)C1)O2 c1(C(=O)NCC(C)N(C)C(c2ccc(F)o2)=O)c(Cl)cc(Cl)cc1Cl N1(Cc2cccc(N(C)CCO)c2)CCC(C)(CNC(c2nccs2)=O)CC1 C(CCOCCO)(C(=O)NC1CC(O)(CO)C1)NC(C1CCC(F)(F)C1)=O C1(C(=O)NCC(C(=O)NC(c2ccnc(O)c2)C)N(C)C)CC2CCC1C2 c1(COC)cccc(C(N2CC(NC(=O)C(Cl)=CCl)CC2CO)=O)c1C c1(C(N2CC(C(N)=O)(CNC(C(C)OCC#C)=O)C2)=O)ccc2nc[nH]c2c1F c1(OC)cc(OC)c(OC)cc1C=CC(c1cccc2scnc12)=O N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(=O)CCCN2C(=O)CCC2=O)C2CC12 Cc1cccc(C2(NCC(N3CCC(O)C3)=O)CCC2)c1 Cc1ncn(C)c(=O)c1C(=O)NCC1CN(C(C2(C#N)CC3(CCC3)C2)=O)C1 C1(C2CCCCN2C)(NC(n2c(C(CC)C)no2)=O)CCOCC1 CC1(C)CN(C(C2CC23CC3)=O)CC(CNC(=O)Cn2ccc(=O)n(C)c2=O)O1 N1(C(C(C)OCc2cccnc2)=O)CCC2CN(C(C3(CO)COC3)=O)CC12 CC(CCC(=O)NC1CC(NC(=O)CC2CN(C)C2)C(O)C1)N(C)C C1(C(=O)NC2CC(CC(N3CCN(C)CC3CO)=O)C2)Cc2ccccc2O1 CCCCC(C)C(=O)N1CC2(C1)CN(C(c1ccc(NS(=O)(=O)CC)cc1)=O)C2 C1(C(=O)NCC(COC)NC(C2CC(O)C(F)C2)=O)CCCC12CCC2 N1(C(=O)C(O)CCl)CCCC2(C1)CN(c1ccnc3cc(Br)nn13)CCO2 Cc1cc(OCC(O)CNC(Cc2nncn2C)C(=O)O)cc(CN)c1 C1(C(=O)NC2(CF)CCN(C(=O)CCc3scnc3C)C2)(OC)CCSCC1 C(=O)(CC(C)C(C)(C)C1CC1)N1CCN(CC)C(=O)C1.C12CC(C1)NC(=O)C2 N1(C(CC(=O)NCC)=O)CC2COCCC2(NC(=O)Cc2ccc(F)cc2C)C1 N1(Cc2ccc(C(N)=O)cc2)CC2(CCOCC2)C1.c12ccc(s1)C(=O)NC2 Cc1cnn(CC(=O)NC2CCC(NC(c3cscn3)=O)C2)c1 c1(C(=O)NC2C(NC(C=C(C)C(F)F)=O)CC2)ncnc2c1CCC2 C1(C(=O)NC(c2ccccc2)CNC(C2(CO)CCC2)=O)CN2CCN1CC2 CCCCC(C)CC(=O)NC1C=CC(C(=O)NC(C)CCC)C1 Cc1nc(O)c(C(N2CCC(CNC(C3CC4CCC(C3)C4F)=O)C2)=O)nc1C n1(CC(=O)NC2CCC(CNC(C3C(OC)CCC3)=O)C2)ccc(=O)cc1C C=CC(C)(CC)C(=O)NCC1(F)CCN(C(c2ccc(C)c(F)c2)=O)C1 C=CCCCCCN(C)C(C1CSCCN1C(=O)Cc1cc(C)no1)=O C(=O)(CCCCC(F)(F)F)N(CCN(C(=O)C(C)C1CCCC1)CC)CC C12(C(N(CCCCO)CC)=O)CCN(C(c3nc(O)sc3C)=O)CCC1C2 c1(C(=O)NCC(CC)NC(=O)CNS(=O)(=O)N(C)C)cccc(Cl)c1C c1(C(N2CCC(F)(C(C)C)C2)=O)cccc2nccn12.C12(CCCC1)C(=O)NC2 c1(C(=O)NC(C(C)NC(C2(CC#C)CC2)=O)C)ccc(OC)cc1 C(C1=NOC2CCCC12)NC(C(C1CN(C(CCC=C)=O)C1)O)=O C1(CC(=O)NCC2(C(C)NC(c3cccc(OCN)c3)=O)CC2)OCCOC1(C)C C(=O)(C(C)(C)CCF)NCC(C1(O)CCN(C(C23CCOC(C)(C2)C3)=O)C1)C c1(CN(CCC(=O)NCC2CCN2C(=O)CCOCCO)CC)ccccc1Cl C1(C(=O)NC(c2nc(C(N3CCC3CC(C)C)=O)co2)C)(CO)CC=CC1 c1(OC)ccccc1-c1ncc(C(=O)NC2CC2CNC(C2CCCN2C)=O)s1 CC(C)(C)C(CNC(C1CC2(C1)CC2F)=O)NC(c1ncn(-c2ccccc2)n1)=O N1(C(C(c2ccc(Cl)cc2)C)=O)CC2(C1)CN(C(=O)C(C)(C)S(C)(=O)=O)CCO2 C#CC1(NC(=O)C(C2(O)CN(C(C34CCCN(CC3)C4)=O)C2)F)CCC(C)(C)C1 c1(OCCOC(C(Cc2ccoc2)NC=O)=O)cnc2ccnn2c1 N1(C(COCc2nc(C)sc2)=O)CCC(C)C1CNC(=O)CCc1cc(Cl)no1 CCCC(O)C(=O)N(C1CCC(NC(=O)C(C)(F)F)CC1)C CC1CCCC2CN=C(NC3CCS(=O)(=O)C3)N12 c1(C(CC)=O)cnc(Cl)[nH]c1=NC(=O)C(C)C1CCOC1 c1(N(C(CNC(C(=Cc2cccs2)C)=O)C)C)ncnc2[nH]ccc12 C12(C(N3CC(CNC(CCNC(=O)OC)=O)C3)=O)CCCCC1CCCC2 CCC(C)CC(C)C(=O)N1CC(C)(C)CC1CNC(c1ccoc1Br)=O c1(CC)nn(C)c(NC(C2CCCCN(C(=O)CC(=O)OC(C)(C)C)C2)=O)c1Cl CCC(CCC(=O)NC1CC1NC(c1ccccc1-c1nnc(C)n1C)=O)OC CCCN(OC)C(=O)CC(CCC)NC(=O)C(N)CCCC(C)C C(=O)(C(C)(C)C(C)C)NCC1CC(Nc2c(C(=O)OCC)cccn2)C1 Cc1c(C(N2CC=CC2CNC(=O)C(F)C(F)(F)F)=O)oc2ccc(F)cc12 C1(NC(C(C)CCN(C)C)=O)CC1C1CCCN(C(C23CCCCC2OCC3)=O)C1 Cc1n[nH]cc1CN(C)C(c1ccoc1CNC(C12CSCC1C2)=O)=O C1(NC(c2nc(COCC)sc2)=O)CCN(C(C2(CC)CCC2)=O)CC12CCC2 c1(C(N(C)CC2N(C(C(CC)CO)=O)CCC2)=O)ccnc(OCC)c1F C(CC(CC)C(=O)N1CC(CC(F)C(N2CC3COCC3C2)=O)C1)=CC C1(NC(CS(=O)(=O)N(CC)CC)=O)CC2CN(C(c3c(Cl)cnn3C)=O)CC2C1 Cc1nc(C(N2CCCC2CN(C(=O)CNC(=O)C2CC2)C)=O)nn1C c1(C(C)CC(=O)NC2CC(C)(NC(=O)C(F)C(C)C)C2)c[nH]c2ccccc12 c1(CC)ncc(C(N2CCC(NC(c3csc(C(C)C)n3)=O)CC2C)=O)c(C)n1 CC1CN(C(=O)C(c2cnn(C)c2)NC(c2ccc(F)cc2)=O)CCN(C)C1 N1(C(c2c(OC)ocn2)=O)CCSCC1C(N1CCC1C1CCC1)=O C(C(CO)(CO)NC(C1(CC2CC2)CC1)=O)N(C)CC1OCCC1(C)C c1(CC)ccc2c(c1)CCC2N=c1[nH]c(=NC)c2[nH]ccc2[nH]1 c1(CC)nc2sc(C)cn2c1C(=O)N(CCCCCNC(=O)CN(C)C(C)=O)C C1(NC(c2ccc(OC)s2)=O)CN(C(c2coc(CO)c2)=O)CC12CCOCC2 CC(CC(N)=O)C(=O)N1C(C(=O)NCCCc2nncs2)CC2CC12 C(C)(CCCCNC(c1cccc(SC)n1)=O)NC(C1(CC#C)CCOC1)=O N1(C(CCOCC)=O)CC2CC(NC(c3ccnc(SC4CCC4)c3)=O)CC1C2 N1(C(C(COC)O)=O)CCN(C(c2ccn(C3CC3)n2)=O)C(C(F)F)C1 n1(CC(=O)NCC(C(C)C)NC(CC(CC)C)=O)cc(F)ccc1=O c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1c(Cl)cnn1C)=O N#Cc1c(NC(C2CC23CCN(C(C2CCCOC2)=O)C3)=O)cccc1F N1(C(CC(C(C)C)O)=O)CC(C)CN(C(c2cnc3n2CCOC3)=O)CC1C N1(NC(C)C(=O)NCC(C)NC(C2(C)COC(=O)C2)=O)CCN(S(C)(=O)=O)CC1 c1(C(N(C(C)CCNC(=O)CSCC(N)=O)C)=O)ccc(-c2cnco2)cc1 C(=O)(C1=CC2CCCC12)NCC1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 C1(CCOC)CN(C(=O)C2=NOC(C(C)(C)C)C2)CCN1C(=O)CS(N)(=O)=O C1(C(N2C(C(CC)C)CCC2)=O)CC2CCC(C1)N2C(=O)Cn1nccn1 N1(CC(=O)NC(CNC(C(CC)F)=O)(C)C2CC2)CCN(C)CC1 c1(C(N2CCCC(NC(C3CC4CCC3O4)=O)CC2)=O)cc2c(nn1)OCCS2 c1(OCC)nc(N2CCC(O)C(C(=O)NCC3CC(=C4CC4)C3)C2)ncc1Br Cc1ccc(C(=O)OCC2CC=CCC2)nn1 C1(NC(C2C(C)N(C(C3CC3c3ccco3)=O)CC2)=O)CC2(CCCCC2)C1 Cn1c(C(=O)NC2CC(NC(C3(CO)CCCO3)=O)C2)cnc1O CC(O)C(C(=O)NCCC1(C)CC1)NC(C1CC1C(C1CCC1)=O)=O c1(C(=O)NC(C(=O)N(C2C(C)CCC2)C)CN(C)C)cc(Cl)ccn1 C1(NC(Cn2cc[n+](C)c2)=O)CSCCN1C(=O)CCOc1ccc(Cl)cc1 c1(C(=O)NC2C(NC(c3c(CC)nn[nH]3)=O)CCC2)c[nH]c2cccc(Cl)c12 C(=O)(C1=CNS(=O)(=O)N=C1C)N(CC(C)O)CCNC(C(C)OCC#C)=O C1(C(N2C(CNC(C3C(C)(C)C3C#N)=O)CCC2)=O)CC(=O)CC(=O)C1 C1(NC(CCc2ccn(C)n2)=O)CN(C(C2CC2c2cnn(C)c2)=O)CC1F Cc1ccc(CC(=O)NC2CCN(C(c3cc(O)nc(Cl)c3)=O)CC2F)c(C)c1 c1(C(=O)NC(CC(C)C)(C)CNC(C2CC=CCO2)=O)ccc2cncn2c1 O=C(C1=Cc2ccccc2C1O)NC1C=CCN(C(c2csc(Cl)c2)=O)C1 N1(C(CN2CCC(OC)C2)=O)CC2(C(=O)NCCCCCCOC)CC1CO2 N1(C(COCC(C)C)=O)CCCC(CN(C)C(c2cc(C(N)=O)cn2C)=O)C1 c1(C(=O)NCCC(C)N(C(=O)CC2(C)CC2)C)ccn(C)n1 Cc1cc(C(=O)NC2CC(O)CN(C(c3ccccc3C(C)C)=O)C2)cc(C)c1 N1(C(c2cnc(N(C)C)c(Cl)c2)=O)CC2(COC(CNC(C3C=CCS3)=O)C2)C1 C1(CC(=O)Nc2ccc(NC(C3C(=C)C3)=O)cc2C)CCc2ccccc2C1 C1(C(=O)NC(C)CC2CCC2)CCCCN(C(C2(C#N)CCCO2)=O)C1 c1(CC(=O)NCCC2CCN(C(c3ccc(C(F)F)s3)=O)C2)nnc2n1CCCC2 c1(N2CCC(CO)C2)nc2ccsc2c(=NCc2ccsc2Br)[nH]1 C1(NC(Cc2cc(CC)no2)=O)CC2(C1)CC(CNC(=O)C(C)C(C)C)C2 c1(C(N2CCOCC(CNC(CS(=O)(=O)NC)=O)C2)=O)c(C)cc(C)cc1C c1(C(N2C(CCNC(C(C)(C)F)=O)CCC2)=O)cnc2cc[nH]c2c1 CCCC(O)CC(=O)NCC12CC(NC(=O)CSc3n[nH]c(O)n3)(CO1)C2 CCN=C(NCc1cnc(Cl)c(C)c1)N1CCC(O)C1 C(CCC(C)NC(c1cccnc1)=O)NC(C(c1ccccc1)C)=O c1(C(C)C)cc(NC(C2CCN2C(=O)COCC2CCCO2)=O)ns1 C1(C(=O)NCC(CC)C(C)(F)F)N(C(=O)CN(C)CCOC)CCCC1(C)C C=Cn1nncc1C(=O)NC(COCC)C(=O)NCCC1COCCO1 N#Cc1ccc(C2(NC(=O)NCc3nonc3Cl)CC2)cc1 CN1CCC(CC(=O)NC2CCN(C(C3(N4CCCCC4=O)CC3)=O)C2)CC1 c1(NC(c2ccnn2C2CNC2)=O)ccc2oc(Cl)cc2c1 Cc1ccc(C=CC(=O)NC(C2(O)CN(C(C3CCC(=O)N3)=O)C2)C)cc1C Cc1cc(C(N2CCC(C(C)NC(=O)CC(c3cccs3)C3CC3)C2)=O)c(C)s1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(C(C)NC(C2(C(C)(F)F)CC2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NCC1CCN(C(C(Cc2ccccc2)N(C)C)=O)C1 C(CNC(=O)CCc1cscn1)(CC(F)(F)F)NC(C(C1CC1)OC)=O c1(CC(C(=O)OC)NS(=O)(=O)CC2CCOC2)cc(Br)sc1Br C1(NC(c2c(COC)scc2)=O)CC2CCC(C1C)N2C(=O)Cc1cc(C)on1 c1(CC(=O)N(CC(O)CN(C)C(C2CCCC2)=O)C)cncnc1O N1(C(CC2(C=C)CCC2)=O)CCC(C2CC2)C1CNC(C1C2C3CCC(C3)C12)=O C1(C)(NC(C=CC(C)NC(C2CC3CC3C2)=O)=O)C(C)(C)C1(C)C c1(C(CC)C)nc(C)c(CC(=O)NC(C)CCCNC(=O)C(C)C#N)c(C)n1 C1(CC(=O)NC(C2CCN(C(CCCOC(C)=O)=O)CC2)C)CC(O)C12CCC2 O=Cc1cccc(-c2nc(Cc3cccs3)no2)c1Br C1(C(N2C(C)(C(=O)NCC(CCOC)O)C=CC2)=O)CC2(CCC2O)C1 CCCC(C)(C)CC(=O)N(C1CCN(C(=O)CC2(C)CCCO2)CC1)CC1CC1 c1(C(N2CCCC(F)(CNC(=O)C=CC=C(Cl)Cl)C2)=O)nc(O)nc(O)c1F c1(C(=O)NC2C(CNC(C(CC=C)(C)O)=O)CC2)cc(C)c(F)c(C)c1 C(=O)(CCC(C)(F)F)NCC(CC)NC(=O)CCNC(=O)CO N1(C(CNC(C)=O)=O)CCC2C(NC(=O)Cn3cccc3)C12 c1(C2(OC)CCN(C(c3n(CC)ccn3)=O)C2)cc(Br)ccc1F C(=O)(CC(O)C(C)C)N1CCC(OCCNC(c2nc(C)c(C)s2)=O)CC1 N1(C(CC=C(C)C)=O)CC2CCC1C1CN(C(c3c[nH]nc3C(F)F)=O)CC21 N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CCN(C(=O)C=CI)C2 CCC(O)C(C)(C)C(=O)N1CCC(N(C(c2cc(N)ccc2Cl)=O)CC)C1 c1(C(=O)NC2C=CC(CC(N3CCC(OC)C3)=O)C2)nccc(C)c1N CCC1(CNC(c2cn(C3CC3)cn2)=O)OCCc2ccccc21 C=CCC(C(=O)NCCCCN(C(=O)Cn1nccc1C)CCO)NC(C)=O N1(C(C(CC)(CC)OC)=O)CC(NC(=O)CCCCCOC)C(C2CC2)C1 Cc1cccc(C(O)C(=O)NCC(c2ccccc2)NC(C2CCCN2C)=O)c1 N1(C(c2c(C)noc2)=O)CC2CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 C(CCC(=O)NCCC1CC(NC(C2CCC=CCC2)=O)C1)NC(N)=O CC(C)(CCCNC(c1sccc1F)=O)NC(=O)COc1ccccc1C(N)=O c1(CC)nsc(CNC(=O)C(C)CN(C(=O)CCc2cc(C)no2)C)n1 N#Cc1ccc(C(=O)Nc2ccc(SCc3nc(=O)o[nH]3)cc2)nc1 C(=O)(C1Cc2ccc(Cl)cc21)NCCS(N=S(C)(C)=O)(=O)=O CCCCC(COC)N=c1nc2c(ncn2C)c(NCc2ccc(Cl)c(Cl)c2)[nH]1 c1(C(=O)NCC(C)N(C(=O)CCNc2ccccc2)C)cc(S(N)(=O)=O)cn1C C(=O)(C(C)(C)C(=O)NCC1CC(C)(C)CN1C(=O)C(CC(C)C)N(C)C)NC CN1C(=O)C2=C(N(c3ccsc3[N+](=O)[O-])C(=O)NC2c2ccn(C(F)F)n2)C1(C)C Cn1cnc2nc(=NCCC3CCN(C(c4coc(CO)c4)=O)CC3)[nH]cc12 C1(COC)(NC(c2cc(Cl)cnn2)=O)CCN(C(=O)CCCc2ccccn2)C1 C(=O)(C(=O)CCC(C)C)N1C(CCOC)CN(C(C2CCOC2C(C)C)=O)CC1 C1(CC)CN(C(c2cc(C)ccc2I)=O)CCN1C(c1cnc(Cl)s1)=O C1(NC(=O)Nc2cnn(-c3nc4ccccc4[nH]3)c2)CCc2[nH]nc(O)c2C1 c1(C(=O)NCCC2CCN(C(C3CC(CF)C3)=O)C2)cccc2cc(Cl)ccc12 c1(C(CNC(c2cc(Cl)ns2)=O)NC(=O)C(O)CF)ccc2ccccc2c1 C(CCN(C1COC1)N1CC(n2cnnc2)C1)OCCOC.C(C)OC c1(OC)cc(Br)ccc1CN1CC2CC1CN2Cc1ccc(C(=O)N(C)C)nc1 C#Cc1ccc(OC)c(C(=O)NC2COCC2NC(c2conc2C2CC2)=O)c1 C1(CC(=O)NCC(=O)NC2CC(CNC(c3cncnc3)=O)C2)CCOCC1 C1(CC(=O)N(CC(=O)OC)CCOC)CCC12CCOCC2 C#CCCCCC(c1nnnn1C)Nc1c(C(C)C)cccc1C C1(c2ccccc2)(NC(C2C(C(=O)Nc3n(C)ncc3)C2)=O)CCOCC1 C1(NC(c2cc(OC)no2)=O)CN(C(C2CC(C)C2)=O)CC1N=[N+]=[N-] C12(CNC(c3cnn(C)c3Cl)=O)CC(C1)C(NC(=O)C(O)c1ccsc1)CO2 CN=c1[nH]c(=NCC(C)SC)[nH]c(=NC2CCC(N3CCCC3)CC2)[nH]1 Cc1cc(C(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)ncc1F c1(C(N2CC(OCC)(CNC(c3cc(F)c[nH]3)=O)C2)=O)cccc(C)n1 c1(C(N2CC(NC(C3(O)CCOCC3)=O)CC(O)C2)=O)cccc2ccccc12 C(=O)(C(C)CC(=O)OC)NCCCN(C(c1ccc(Cl)o1)=O)CC Cc1nc(S)nc(C)c1CCC(=O)NCCCN(C)C(c1ncccc1Cl)=O c1(C(N2CCCC(F)(CNC(C(COC)C)=O)C2)=O)cnc2c(c1)NC(=O)CO2 C1(CNC(C=C(CNC(C(C2CCCC2)OCC)=O)C)=O)CC(CO)CO1 N(C1COc2ccccc21)C(=O)NCCCOC1CCOC1 c1(NC(C2CC(C(=O)NCCCOC)C2)=O)c(C)nn(-c2ncccc2Br)c1C C(c1cnc(C)nc1O)=CC(=O)NC1CCN(C(c2occ(C)c2)=O)C(C)C1 C(=O)(C(=O)N=S(C)(C)=O)N(CC(CN(C(=O)CCC(=O)c1ccc(Cl)s1)C)O)C c1(OC)ccc(Cl)c2c1CN(C(c1nccc(C)n1)=O)CC2 CN1CCC(CO)(CNC(=O)C(CCC2CCC2)NC(=O)Cc2nccn2C)C1 c1(C(=O)NCC(C)N(C(=O)CCc2cccnc2Cl)CC)c(C)cccc1C c1(CCC)ccc(C(=O)NCc2cc(C(N3CCCC3CC)=O)on2)s1 C1(NC(c2ncoc2-c2ccon2)=O)CCCC(CNC(C2CC(O)C2)=O)C1 c1(C(=O)NC(C(=O)NCC2OCC(C)(C)C2)C2(O)CCC2)cc2ccccc2o1 c1(C(N2C3C(NC(=O)C=CC=C(Cl)Cl)C(CC3)C2)=O)cc2c[nH]cnc-2n1 N1(C(CC2(C)CCC2)=O)CCC(O)(CCNC(c2ccc(F)cc2)=O)C1 C1(NC(c2scc(CC)c2)=O)CCOCC1C(=O)NCC1(OC)CCCCC1 C(=O)(C1=Cc2ccccc2C1)NCC(CNC(C1CC(C)(C)OCC1)=O)CO CCCCC(=O)C(=O)N1CC(CC(=O)Nc2ccc[n+]([O-])c2)C(C)C1 CC1CC(CO)CN1C(=O)C#CCNC(=O)CCCC1CCCO1 Cc1nn(C)cc1NC(c1cncc(CNC(=O)CC2CCCCC2C)c1)=O c1(C(C)(F)F)ccc(C(=O)NCC(C)(O)CNC(C2CCCO2)=O)cc1 C1(NC(=O)NC2(OCC)CCCC2)C2CN(C(C3C4CCC3CC4)=O)CC12 CCC(C)(CO)C(=O)NCCC1CCN(C(c2csc(=N)[nH]2)=O)C1 C(CCO)OC(C)=O.S(C)(=O)(=O)N(CCN)C(C)C1CC1 c1(C(=O)NCCN(c2ncc(C)c(C)n2)CC)sc2nccn2c1C N1(C(C(CCOC)C)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 c1(C(=O)NC(C)CN(C)C(C2(Cl)CC2(F)F)=O)nc2c(s1)CCCC2 c1(CNC(C(C2CCCOC2)OC)=O)cccn1C(c1ccncc1)C C(=O)(C(C#N)(CC)CC)N1C2(C(N3CC(C#C)C(OC)C3)=O)CC(C1)C2 Cn1nc(C(=O)NCC(C)(Cn2cccn2)NC(=O)CNS(N)(=O)=O)cc1O CC1=NOC(=O)C1CC(=O)NCCC(C)NC(=O)Cc1nc(C2CC2)cs1 C(CC(N)=O)(C(=O)NCc1cn(C)nc1O)NC(CCC=C=C)=O c1(CCC(N2CC(CCNC(=O)C(C3CC3)SC)(OC)C2)=O)cccnc1F O(NC(=O)CCCC(C)(C)NC(=O)C(C1CCC1)OCC)CC(=O)OC C(CN=C(NCc1ccsc1)NC(C)C1CC1)c1ccc(SC)cc1 c1(C(=O)NCC2N(C(CCC3CC(OC)C3)=O)CC2)ncccc1O c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CCOC2)cc(=N)[nH]c(Cl)n1 c1(C(N(C2CC(NC(=O)CCCC#N)C(O)C2)CC)=O)cnc2[nH]cc(C)c2c1 Cc1cc(C(N2CCC(c3nncs3)C2)C(=O)NC2(C)CC2)cs1 c1(C(N2CC3(CC(NC(C(C)(C)SC)=O)C3)C2)=O)ccc2n[nH]cc2c1F c1(C(N2CC(NC(C3CC3(Cl)Cl)=O)CC(OC)C2)=O)ccc(C#N)c(C)c1 Cc1ccn(C(C)C(N2CCC(CCC(=O)NC(C)(CO)C3CCC3)C2)=O)n1 N1(C(C(C=C)O)=O)CCN(CCNC(c2cn(C)nc2C)=O)CC1 N1(C(CC=C(C)C)=O)C(C(=O)N(C)Cc2ncc(C)o2)CC2CCCC12 c1(C(=O)NC(C2CCCN(C(c3cc(F)n[nH]3)=O)C2)C)ccc2nsnc2c1 C(=O)(CS(=O)CCC(F)(F)F)NC(C1CCCN1C(c1cc2cccnc2s1)=O)C C1(NC(CCC)=O)CCC2(CCCN2C(c2cccn(C)c2=O)=O)CC1 N1(C(c2c(CC)c[nH]n2)=O)CCCC2(C1)CN(C(=O)CN1OC(C)(C)CC1=O)C2 C#Cc1cccc(NC(=O)C(C)NC(=O)CCC(C)SCC)c1 N1(C(C(CC)NC(N)=O)=O)CCOCC2(COCCN2C(=O)C(F)C(C)C)C1 c1(C(=O)OC)cc(NC(=O)C(=O)Nc2ccc(SCC(C)C)cc2)c(C)cc1F c1(C(=O)NC(CN(C(CC(c2ccc(F)cc2)C)=O)C)C)ccc2ncnn2c1 c1(C(N2CCN(C(C(c3c(C)cncc3)C)=O)CC2)=O)cc(Br)cc(N)c1C Cc1ncc(NC(=O)C(C2CCCN(C(C3CN4CCC3CC4)=O)C2)C)c(C)n1 c1(N2CC(C)C(N3CCOCC3)C2)cc(Cl)c(I)cn1 c1(C(=O)NCC2(CNC(C(C)Cn3cccn3)=O)CC2)ccsc1C#N CC1C(NC(c2ccc([N+](=O)[O-])s2)=O)C(C)CCN1C(=O)Cn1cccc1 CC1(C)COC(CNC(=O)C(C2(C)CC2)NC(=O)CC2CC(F)(F)C2)C1 N1(Cc2c(OC)nccc2)CCCN(C(=O)CNC(=O)N(C)C)CC1 C(=O)(CC(F)(F)C(C)C)NC1CCC(CCNC(C2(OC)CCSC2)=O)C1 C1(NC(C(CC)(F)F)=O)CCC2CC1CN2C(=O)C(=Cc1ccccn1)C CC1CN(C(=O)CCC2CCCN(C)C2)CCCN1C(=O)Cn1cccnc1=O C(CC1=CCOCC1)N(C(=O)CCNC(=O)CN1CSCC1=O)C c1(N(CC(=C)C)CC)nnc(C(C)C2CC2)n1CCCCCC CN1CCOCC1(c1cn(CNC(c2ccc(NC3CCC3)cc2)=O)nn1)CO C1(NC(C(C)C2CC2)=O)C=CS(=O)(=O)C1.C12(NCCO)CC(C(=O)N)(C1)C2 c1(C(=O)OC)ccc(NC(=O)NC23OCC(C(COC)C)(C2)C3)cc1.C(C)(C)(C)O C1(C(=O)NCC(C)NC(C2(CC=C)CC2)=O)CCn2ccnc2C1 C(=O)(C(C)(C)C)NC(C(=O)NC(C(=O)N(C1CC(F)(F)C1)C)CO)CC1CCC1 C1(CCNC(C2(C(CC)=O)CC2)=O)C(C)CCCN1C(c1coc(O)n1)=O c1(C(=O)NC(CC(C)NC(=O)C=CI)C)c(Cl)cnn1C c1(CC(=O)NCCNC(C(C)Cc2ccc(Cl)cc2)=O)c(O)ncnc1O c1(C(=O)NCCCCCNC(c2ccccc2C(F)(F)F)=O)cc2n(c1)CCC2 n1(CCOC)cc(C(=O)NCC2(C(C)(C)O)CN(C(C3CC4CC4C3)=O)C2)cn1 c1(NCCC(C)(C)NC(C2N(C)CCOC2)=O)ncnc2c1COC2 N1(C(C(CC2CCC2)OC)=O)CC(F)(F)CC1CNC(c1cc2n(c1)CCC2)=O c1(C(=O)NC2(C)CC(NC(c3c(CC)c[nH]c3)=O)C2)cc2c(Br)cccc2[nH]1 N1(C(CNSSC)=O)CCCC2(NC(c3cccc4oncc34)=O)CCCC12 CC(N=c1cc2n([nH]1)CCNC2=O)c1cnc[nH]1 C1(NC(=O)CCN2CCCC2)C=CCN(C(=O)CNc2ccc(O)cc2)C1 Cc1cc(OC(F)F)nc(N2CCCC2CO)n1.C12CCCN(C1)C(=O)CN2C C1(NC(C(CC=C)C(C)C)=O)COC2(CCN(C(c3sccc3Cl)=O)CC2)C1 C(C1=CCN(C(c2scnc2Cl)=O)CC1)NC(C1C(C)C1C)=O c1(C(N(C)CC2N(C(CC=C)=O)CCOC2)=O)c[nH]c2ncnc(O)c12 C12(NC(C(CC(C)C)O)=O)CCCCC1CN(C(c1nc3cnccc3s1)=O)C2 c1(C(=O)NC(C)CCCNC(=O)C(O)C2CCC2)cnc2sccn12 N1(C(c2cc(C#C)cc(Br)c2)=O)CCC2CN(C(=O)CCC(F)F)CCC12 C1(NC(c2n(C)c(S)nn2)=O)CC2CCC1N(C(c1ncc(F)cc1F)=O)C2 C1(NC(C(CO)OC)=O)CCCCCN(C(=O)C(C)O)C1 N1(C(C2CCC3(CCC3)CC2)=O)CC2CCC(C1)N2C(C12CCCC1C2(F)F)=O c1(CC(=O)NC(CN(C(CSCCOC)=O)C)C)c(O)ncnc1O Cc1c(C(=O)NC2CC(C)(CNC(=O)CCCCN(C)C)C2)cccc1O C#CCCCCCC(=O)NCC1(C)CCC(C(C)(C)C)CC1 C1(C)(C(=O)NC2CCCCN(C(c3c(CC)non3)=O)C2)CC2(CC(O)C2)C1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CCCC(NC(=O)C(F)(F)c2ccnn2C)C1 CC(C)(C)C(O)C(=O)NC1CC(NC(c2cc(C(F)F)cs2)=O)CC1O C(CC(CC)C(=O)N1CC(C(=O)NOCC(C)(C)C)CC(C)C1)=CC N1(C(C2CNCCN2Cc2cscn2)=O)CC2CCCCC2C1 C12(NC(C(C(C)C)Oc3cccc(Cl)c3)=O)CCCC1CN(C(=O)C=CCF)C2 c1(C(N2CCN(C(C(C=C)O)=O)CC2C)=O)cc(Br)cc([N+](=O)[O-])c1C c1(CNC(=O)C(N2CC(F)(F)CC2c2ccccc2)=O)c(O)ncnc1O C1(C(=O)OC)CC(C)N(C(=O)NCCC(C)SC(C)(C)C)C(c2ccco2)C1 C1(N)CCCCC1C#N.N12CCN(CC1)CC(=O)NCc1ccoc1C2=O.CO c1(C(N2CC(CNC(=O)CCCc3nccs3)C3C2C3)=O)ccc(O)c(Cl)n1 C(CCSC)(C(=O)NC(C)CCC)NC(CCC#C)=O c1(CNC(C2C(NC(=O)CC34CCCC3C4)COC2)=O)cccnc1Cl C1(CNC(c2c(CC)c[nH]n2)=O)C2CN(C(=O)CC3CCC(=O)CC3)CC12 S(=O)(=O)(c1cc(Cl)c([N+](=O)[O-])cc1F)Nc1c(CC)cccc1C(=O)OC CC(C)S(=O)(=O)CC(=O)N1CC(F)(CNC(=O)CC2CCCCC2(C)C)C1 CCC(Cc1ccccc1C)C(=O)NC1CCCCC1NC(c1nsnc1O)=O N1(C(COCC(=O)OC)=O)CCCC(N(C(=O)CCN(c2ccccc2)C)C)C1 C1(CNC(CN(CCC#C)C)=O)CN(C(=O)C(O)CCSC)CC1F c1(C(N2CCC(O)(c3cn(C(C)C)nn3)C2C(=O)O)=O)cccn2nccc12 C(=O)(C(F)CC(C)(C)NC(c1cccn2ccnc12)=O)N1CCCC(C)(CC)C1 N1(C(c2c[nH]c(=NC)o2)=O)CCCC1C1CCCCN1C(=O)CN1CCCCC1 C1(C(=O)NC(c2cncn2C)C)CCC(O)CN1C(c1cnc(S)nc1)=O C1(C)(C(=O)NCc2ccc(C3C(C)C3)o2)CCCN1C(c1ccsc1C#N)=O CC1CC(NC(=O)C2=NNC(=O)C2)CN(C(c2cc(=N)[nH]c(=N)[nH]2)=O)C1 c1(C(N(C2CCN(CC)CC2)c2n(CCC)ncc2)=O)nc(C)c(C)n1C N1(S(CCOCC)(=O)=O)CC2CN(C(c3cnn4c3CCCC4)=O)CC2C1 N1(C(C2C(C(=O)OCC)CC2)=O)CC(NC(C2CC2c2ccccc2)=O)C(O)C1 C1(NC(CS(=O)(=O)N(CC)CC)=O)CC2(CCN(C(=O)C(C)=C(C)C)C2)C1 C(C(CC(=O)N1CCC(NC(c2cc3occc3n2C)=O)C1)C(F)(F)F)N(C)C c1(C(N)=O)ccc(C(=O)N(CCNC(C2CCCC2C(F)F)=O)C2CC2)o1 C=CCC(C(=O)NCC)NC(=O)OC(C)(C)C.C1(=O)C(COCCO)N1C.NC C1(N(C)C(C2COCCO2)=O)CCC(NC(c2sccc2C#N)=O)CC1 N1(C(=O)Cn2nnc(C3CC3)n2)CCC2CCN(C(C3C4COCC34)=O)C2C1 N1(C(c2cc(C(=O)NCC)no2)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 c1(SC(C)C(=O)OC(Cc2cccnc2)C(F)(F)F)c(F)cccc1Cl C1(C(=O)NC2CC(CNC(C(CN(C)C)(C)C)=O)C2)CCC(N=[N+]=[N-])CC1 C12(CCCC1)C(C)(NCC1CC(C)C1)c1nnnn1CC2.c1(CO)nnn(C)n1 Cc1nc(O)ccc1C(=O)NCc1cc[nH]c1C(=O)N(CCCCO)C1CC1 C1(CC(N2CC(NC(c3nc(C)oc3)=O)C(C)C2)=O)OCCCC1(C)C O=S(=O)(Nc1cnn(-c2ccc(Cl)cc2)c1)N1CCC(F)(F)C1 C1(CN(C)C(c2cc(CCCO)on2)=O)CCCN1C(c1ccc(C(N)=O)[nH]1)=O c1(NC(C23C(CN(C(C4(Br)CC4)=O)C2)C3)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C2C(C)(C)COC2)=O)CC2(C=C(C(=O)NCCC34CCCC3C4)CO2)C1 C(=O)(CCCC(=O)NC)NCc1cc(C(N2CC(O)(CC=C)C2)=O)n[nH]1 N1(C(c2cnc(C3CC3)nc2)C(=O)NCCC)CC(N(C)C)C(C)C1 c1(CNC(c2nc(CC)sc2)=O)cc(C(=O)NCC23CCCCC2C3)ccn1 N1(C(CN(C)C)=O)CCOC2CN(C(=O)C=Cc3ccco3)CC12 Cc1ccc2nc(N3CC=C(CCNC(C4OCC4(C)C)=O)CC3)sc2n1 C1(CNC(=O)CCc2ccc(Cl)s2)CCCN(c2ccnc(N3CCCCC3)n2)C1 Cc1cc2nccnc2cc1C(=O)NC(C)CCNC(C1CC2(CCC2)C1)=O C=CC1(CC(=O)NCCC(C)N2CCC2)CN(C(c2nccnc2N)=O)C1 Cc1cnc(N(C2CCCNCC2)C(c2ccc(CO)o2)=O)nc1 CCCCC(O)CC(=O)N1CCOC(CCNC(c2ncc([N+](=O)[O-])n2C)=O)C1 c1(C(N2CC(CNC(CCCCSC)=O)C(C)C2)=O)ccnc(O)c1F c1(CC(C)C)cc(C(=O)NC2(CCNC(=O)CO)CCC2)no1 N(C1CCCOc2ccc(F)cc21)C1CC(C(C)(C)C)OCC1 C1(NC(c2cc(OC)c(C)cc2)=O)CN(C(c2occc2Cl)=O)CCC12CCC2 c1(C(N(C2CCN(c3cc(CC)cnn3)C2)CCC)=O)ccc2c(c1)OCO2 CC1CC(C)(NC(=O)C=CCN(C)C(C2CNC(=O)N2)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NCCC1CC(NC(C2CC23CCCOC3)=O)C1 C1(C2CCN(C(C3CC4CCC3O4)=O)C2)(NC(c2c(C)nc(C)o2)=O)CC1 C1(C(N(C2CCC(NC(c3c(CC)nn(C)c3)=O)CC2)C)=O)CCCC1C1CC1 c1(C(C(=O)NCCCC)N(CCC)Cc2ccco2)scnc1Br c1(C(=O)NCC2N(C(C3C(C=C)CC3)=O)CC(O)C2)cc(Br)ccc1OC Cc1ccccc1CCNC(=O)CC1CC(c2cccc(Br)c2)C1 N1(CC(=O)NC(C2CCN(C(=O)CC3CCOCC3)C2)(C)C)CCSCC1 C(=O)(CCC(CF)CF)N(CC(=O)NCCC1CCOCC1)CC#C C(=O)(CCCC(F)(F)F)N1CC(C)C(CNC(c2nc(Cl)cc(N)c2Cl)=O)C1 CC(CC(=O)Nc1ncc(CCNC(C2(CC3CC3)CCC2)=O)s1)n1cccc1 c1(CC2N(C(n3cc(C(CC)(O)CC)nn3)=O)CCC2)cn2ccsc2n1 c1(COC2CN(C(c3cnc(-c4ccccn4)s3)=O)C2)cccnc1 c1(C(C)=O)oc2ccccc2c1NCCC(=O)NC.C1(C)CCN(C(=O)C(C)CC)C1 C(=O)(C1=CC2C=CC1C2)NCC1C(C(N2CC(C3CC3)(OC)C2)=O)C1(C)C C#CC1CN(C(c2ccc(OC)nc2)=O)CCN1C(=O)CSCC(N)=O N1(C(C=CC(C)(C)C)=O)CCC(F)(CNC(=O)C(O)Cc2ccccn2)C1 c1(C(N(C(C(=O)NCCC(C)SC)=O)C)CN2CCOCC2)cc2ccccc2o1 CC(C(=O)NN1CCCC1C(N1CC(OCC(N)=O)C1)=O)NC(N)=O N1(C(c2cnc(C(C)O)s2)=O)CC2(C1)CN(C(=O)CC1NC(=O)NC1=O)CCO2 C1(NC(C(C)NC(CC)=O)=O)CC12CC(NC(c1cnn(C3COC3)c1)=O)C2 c1(C(=O)NCC(CNC(CCC(=O)NC)=O)C)nc(C)c(C)cc1N N1(C(C2C(OC(C)(C)C)C2)=O)CC2(C1)CN(C(=O)C1=CCCOC1)C2 c1(C(=O)NCC2CC(=C)C2)oc(CNC(c2ccc(CC)s2)=O)cc1C N1(C(C(C)SC(C)C)=O)CCC(F)(CNC(=O)C=Cc2ccc(C(N)=O)o2)C1 N1(C(CC2CC(=C)C2)=O)CCN(C(=O)C(n2cc(C)cn2)C)C(C(C)C)C1 c1(N(C)Cc2c(C)nc(-c3ccccc3)s2)nccc(=NC(C)c2ccsc2)[nH]1 N1(C(C(=O)NC2CC(N(C(c3ncc(OC)cn3)=O)C)C2)C)CCP(C)(=O)CC1 C(c1ccc(N(C)C)cc1)=CC(=O)NCC1(CNC(c2scc(C)c2)=O)CC1 C1(C)(CNC(C(CSC)c2ccccc2)=O)CCN(C(C2CCCSC2)=O)CC1 N1(C(C2C(C)(CC)C2)=O)CC2(CC(NC(C3CC(=O)NC(=O)N3)=O)CO2)C1 C1(NC(c2cc(COC)no2)=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCCC12 C1(C(=O)NC2C3C=CC(C3)C2CO)CC2CCC(C1)N2C(=O)C1=CCCCO1 C1(CC(C)NC(CCOCCCC)=O)CCN(C(=O)C(C2(O)CCCC2)F)CC1 C1(C(N(CC(CC)NC(=O)CSCC(F)F)CC)=O)C2COCC12 c1(C(=O)NCC(=O)NCC(=O)N(C(C)CO)C)ccc(C#N)o1 N1(C(CC2C(C)CN(C(c3cncc([N+](=O)[O-])c3)=O)C2)=O)CC2CN(C)CC2C1 C(C1c2ccccc2CCN1C(C1(OC)CC1)=O)NC(C1CCC(CC)O1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(F)CC3CCCC3)C2)ccc(N=[N+]=[N-])cc1 C1(O)(CCNC(C2CC3CC3C2)=O)CCN(C(=O)C2=CCOC2)CC1 Cc1nc(O)sc1C(=O)NC1(C(=O)NC2CC(C)(O)C2)CC1(C)C C1(C(N2CCC(OCCNC(C3CCC(=O)O3)=O)CC2)=O)CCN2CCOCC12 C1(NC(=O)C=CC(F)(F)F)CN(C(=O)CC=C(F)Cl)CCC1c1ccccc1 NS(=O)(=O)c1cc(C(=O)NC2CCC2NC(=O)C=CC2CCOC2)c(Cl)o1 N1(C(C(C)C2CCCC2)=O)CC(CC(N2CCC(C(C)(C)C)CC2)=O)C2(CC2)C1 Cn1cc(C(=O)OCc2nc(C3OCCO3)cs2)c2cccc(Cl)c12 c1(CC(=O)NC2CCN(C(CC(CC)CN(C)C)=O)C2C)ccn2cncc2c1 C1(CNC(c2c(CC(=O)OC)occ2)=O)CCN(C(C2CCOC(C)C2)=O)CC1 C(C(C(C)C)NC(=O)CC1CCN(C(=O)Cc2cc[nH]c2)C1)NC(C)=O N1(C(CC(CCC)C)=O)CCOC2(C1)CN(C(=O)C1=C(C)OCCS1)C2 C(=O)(C1Cc2ccccc21)NC(C(NOCC(C(C)C)O)=O)c1cn(C)nn1 CC(C)C(O)C(=O)NC(C(=O)N1CCC(CN(C)C)C1)C(C)C C(=O)(C(C)CC(F)(F)F)NCC1(NC(C=Cc2c(C)n[nH]c2)=O)CCCC1 C1(CC)CCC(C)CN1CC(=O)Nc1ccc(N2CCOCC2)c(C)c1 C1(COC)CCCC(NC(=O)C(n2cc(CN3CCN(C)CC3)nn2)C)C1 N1CC(F)(F)CC1CNC(=O)CSC(COCCCNC)=O.N1(CC2CC2)CCCC1 n1(CC(N2CC(NC(c3n(C)ncc3)=O)C(O)C2)=O)cnc2c1CCCC2 CC(O)(C(=O)NC1COCC1C(=O)NC1CCN(S(C)(=O)=O)C1)C(F)(F)F c1(C(=O)NCC(C)CNC(=O)CC2(C)COCCO2)nc2cccnc2s1 c1(CC(N2CCC(CNC(C3CC34CC(F)(F)C4)=O)C2)=O)ccc(F)c(F)c1 C12(C)CCCN(C1)CC(=O)NCC(=O)N2.CCCCS(=O)(=O)COC C(CNC(=O)CC#N)(CC(F)(F)F)NC(C(C(C)C)n1cc(Br)cn1)=O C1(=CC(=O)NCCCN(C(C)C)C(C2CCC(C)C2)=O)CCN(C)C1 Cc1nc(C)n(CC(=O)NCCC2(O)CCN(C(C3(C#N)CCCO3)=O)C2)n1 C12(NC(C3(C)CC(=C)C3)=O)CCN(C(c3cccc(OCC(C)C)c3)=O)CC1C2 N1(C(c2cncc(C#C)c2)=O)CC2=C(C1)CN(C(C1(C)CC1Br)=O)C2 c1(C(N(C2CCN(C(=O)Cc3sccc3C)CC2)CC#C)=O)ccc(C)cc1Cl c1(CNC(N2CCN(C(C3COCCOC3)=O)CC2)=O)cccc2ccnn12 C1(CNC(C2(C(C)=O)CC2)=O)CC2(CCN(C(c3cccn3C)=O)C2)CO1 Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)C(C)NC=O C(=O)(CC(C)C(F)(F)C(F)(F)F)C=O.C(CC(C)C)(C(=O)NCCCN)OC c1(-c2ccc(C)o2)nn(C)cc1CSC1CCCC(C)C1.n12cc(nn1)NC(=O)C2 N1(C(C2CN(C(C)C)C2)=O)CCCC(C)(CNC(=O)CCCN=[N+]=[N-])C1 c1(-c2cn(CCNC(C(C3CCOCC3)C)=O)nn2)ccc2ncsc2c1 CC(CCCC(=O)NCCCC[Si](C)(C)C)NC(c1ccccc1)=O c1(C(=O)NCC(COC)NC(C2C(C)C2(F)F)=O)ccc(C)cc1 c1(OC)ccc(CCC(=O)NCCCN(C(c2occc2C)=O)C(C)C)c(F)c1 CN1CCCCC1CC(=O)NC1C2CN(C(C3CC34CC4)=O)CC12 C1(C)(C(=O)NCCN(C(C(C)OCc2c(C)cccc2)=O)C)CCC12CCC2 c1(CC(N2CC(c3cn(CCCC(=O)OC)nn3)C(O)C2)=O)cc(Br)ccc1C C(=O)(CCC(C)(C)F)Nc1ccc(SCCNC(C2C(C)CCS2)=O)cc1 C1(C(CN2CCCC2(C)C(=O)OC2CC2)OC(C)C)CCC(F)(F)CC1 C1(C(N2C(C(=O)NCC(C)C(C)(C)C)COCC2)=O)CCC(F)(F)CC1 C=CC(CC)CC(=O)N1CCC(C(C)(C)NC(=O)CN2CCC(C)CC2)C1 C(=O)(C(CCC1CC1)NC(=O)Cc1cnoc1)NCCC1(C)CCC1 Cc1cncnc1C(=O)NC1CCC(C(=O)NCC(C)(C)C(N)=O)C1 c1(NC(=O)C(C)(C)C)cc(C)n(C2CCCC2)c1C.C(C1C(=O)O1)OC(C)=O C1(NC(CCc2onc(C)n2)=O)CCN(Cc2cn(C3CCNC3)nn2)CC1.C12CC1(C)C2 CC(C(=O)N1CC(CCNC(C2(Cl)CC2)=O)C1)N(C)C Cc1ccc(N)cc1C(=O)NCCC1CC(NC(=O)CC2CCCC(C)(C)C2)C1 CC1=C(C(c2nnnn2CC2CC2)Nc2ccc(Cl)c(Cl)c2)C(C)(C)CCC1 C1(COC(=O)C(c2ccccc2)C2CCCC2)CCC(F)(F)CC1 c1(C(=O)NCCN(C(Cc2scc(C)c2)=O)CC(C)O)cc(C(F)F)nn1C c1(C(=O)NCC2CCCC(NC(CCCOCC)=O)C2)cc2cccc(F)c2o1 N1(C(CC(O)C(F)(F)F)=O)CCCN(CCO)C(=O)C1 c1(C(N(CCC)CCNC(=O)CC2(C)CC2(Cl)Cl)=O)ccc2ncc(=O)[nH]c2c1 C1(c2onc(C)n2)CN(C)CCN1C(CC1CCC(C)(C)O1)C(=O)NC1CC1 N1(C(c2c(CNC(C3CC(CC)C3)=O)nnn2C)=O)CCCC(N=[N+]=[N-])C1 c1(C(=O)NCC2CC(NC(C(CCC)O)=O)C2)c[nH]c2ccc(Br)cc2c1=N N1(C(c2cc(CC)nn2C)=O)C2CCC1CN(C(C1C(C)(C)C1(F)F)=O)C2 CC1SCCC1N=c1nc2ncn(C)c2c(NCCc2cn(C)nn2)[nH]1 c1(C(=O)NCC(CO)NC(C(CC)N(C)C)=O)cc(C(=O)OC)cc([N+](=O)[O-])c1 C(CC(CNC(c1coc(Br)c1)=O)NC(c1c[nH]c(C(=O)OC)c1)=O)OC C1(NC(C2=C(C)CCC2)=O)CCOC2(CCN(C(c3cc(CO)[nH]n3)=O)CC2)C1 N1(Cc2c(C)nc(C)nc2C)CCS(=O)(=O)C(CCNC(c2cc(C)sn2)=O)C1 c1(CC(C(=O)NC(C(=O)OCC)CC2CC(F)(F)C2)C#N)ccc(C#N)cc1 C1(C(C(=O)NCC2(CO)CCCC2)F)CCN(C(c2nccs2)=O)C1 CC1CCCC(C)N1CC(N1C2(CN(CC(=O)OCC3CCCO3)C2)CC1)=O c1(OC)cc2nc(NC3CCCN(Cc4cccs4)C3)nc(O)c2cc1OC CCC(CC(F)(F)F)NC(=O)CCN(CCCO)C(=O)Cc1ccon1 c1(C(=O)NC(C2CCCC2)CNC(C(CC=C)(C)C)=O)ccc2oc(=N)[nH]c2c1 c1(C(=O)NC2CC(NC(c3n(CC)nnc3)=O)C2)c(F)ccc(C#N)c1F c1(C2(CC(C)(C)C)CC2)cn(CCCC(=O)NCC(c2ccccc2)(C)F)nn1.C c1(C(N(C2CCN(C(c3ccc(OC)s3)=O)C2)C)=O)cnnc(C)c1 C1(CN(C)C)COCCN1C(C1COCCN1C)=O.n12cc(nn1)CNC(=O)C2 C1(C(=O)NCCC(C)OC)CN(C(=O)CCC)CC1(C)C c1(CSCC(=O)NCCCN(C(C=NOC)=O)C(=O)C2CC2)ccc(Cl)cc1 N1(C(C2C(CC)CN(C(c3ccc4cncn4c3)=O)C2)=O)CC2C=CCC(C2)C1 N1(C(c2c(CC(=O)OC)scc2)=O)CC2CCN(C(=O)CCC(C)SC)C2C1 CCC(CCOC)C(=O)N(CC(N1CC2(CC2)C1)=O)C1CCC1 Cc1ccc(OC(=O)C(C)OCc2cn(CC(c3ccccc3)O)nn2)c(Cl)c1 C1(NC(CCc2ccc(CC)cc2)=O)CCN(C(C2CC23CC3)=O)CC1F C12(C(=O)NCC3CC(N(C)CC)C3)CCCCN1CCC2.N12CCC(O)C1C2=O Cc1ocnc1C(=O)NC(c1ccccc1)C(=O)NCC1(CC(C)C)CC1 N1(C(C(n2cc(Cl)cn2)C)=O)CC2CCCC(C1)N2C(=O)C(C#N)CC1CC1 C1(CCNC(C2CC(=O)OC2)=O)CN(C(C2(CO)CCOCC2)=O)CCO1 C1(NC(C2(C)CCCC2)=O)CCN(C(=O)Cc2cccc(N)c2N)CC1F CCC(CC(C)C)C(=O)NC1CC(C)(NC(C2CC2c2ccncc2Cl)=O)C1 CCC(C)(COC)C(=O)N(C)CCOCCN(C(=O)CNC(=O)CC(C)C)C C(=O)(CC1CS(=O)(=O)c2ccccc21)OCC(=Cc1ccccc1)C#N CC1CCC(=CC(=O)NCCOCCCN(C)C(c2cn(CCO)nn2)=O)C1 Cc1cc(C(=O)NC2CC(NC(=O)CCOC3CC3)C(O)C2)ccc1O c1(OCC(=O)N(c2ccccc2O)CC)cc(O)ccc1OC C(C)(C(C)C(=O)NCC(=O)OC(C)(C)C)NC(c1cc(OCC)no1)=O C1(C(=O)OC)CCCC(C(N2CC(OC)C(n3ccnn3)C2)=O)C1 CCCC(C)C(=O)N1CC2C(N(C(=O)CCOC3CCCCC3)C)C2C1 C1(NC(C(N2C(CSC)CCCCC2)=O)=O)CC2(CCC2)C12CCC2 Cc1nc(N2CCCC(CNC(c3ccno3)=O)CC2)c(C)c(Cl)n1 C=CCCCCC(=O)NC12CCC(C1)N(C(=O)C(C)Cc1cnc[nH]1)C2 N1(C(c2c(C)con2)=O)CCCC2(NC(=O)Cc3nc(F)c(F)cc3F)CC2C1 N1(C(C=CC(C)NC(=O)C2=C(Cl)CCOC2)=O)C2CCCC1CN(C)C2 c1(C(N(C)CC2(CNC(=O)Cc3csnn3)CC2)=O)ccn2nccc2c1 c1(-c2nc(CC(C)(C)CO)nn2CC2CCOC2)ccc(F)cc1C(F)(F)F C=CCN(OC)C(=O)C(F)CC(C)(C)NC(c1nscc1C)=O CCC(C)(COC)CNC(=O)CCCCN(C(=O)C(C)N(C)C=O)C.C1(C)CC1 C1(F)(C(N(CC(O)CO)C)=O)CCCN(C(c2cc3n(n2)CCC3)=O)C1 N1(C(CC(C=C)CC)=O)CC(C)CN(C(c2cnn(CCC)c2)=O)CC1C Cc1ccc2ncc(C(=O)NCC3CCC3NC(c3ccnnc3O)=O)cc2c1 CCCC(CNC(C1(C#N)CCC1)=O)C(=O)NC(C(C)C)C(C)C Cc1nn(C(C)C)cc1C(=O)NC1CC1NC(C1CC1C)=O c1(C(N2CCCC(N(C(C(CCSC)O)=O)CC3CC3)C2)=O)cc(N)c(F)cn1 CC1C(NC(=O)C2=CCC2)CCN1C(c1coc(CC2CC2)n1)=O C1(N(C(CC(CCC)C)=O)CC)CC(C(=O)Nc2ccccc2Cl)=CC1O c1(C(N2CC(C)(CCC(N3C(C(C)O)CC3)=O)C2)=O)cc2ccccc2[nH]1 N1(c2ncnc(C)c2Br)CCC2CCC(C1)N2C(c1cn2c(n1)CCC2)=O C1(N(C)C(c2cc(F)n[nH]2)=O)CN(C(=O)C(F)Cc2ccccc2)CC1O c1(C(C)=O)ccc(C(=O)NCC2(CN(C(=O)C(O)C3CCC3)C)CC2)cc1F c1(CNC(c2c(CNC(C(C)=C3CCC3)=O)n[nH]c2)=O)ncccc1C C1(CC)CN(C(c2ccc(CNC(C3CC(C)C3)=O)s2)=O)CC(CC)O1 N1(C(C(CC)NC(N)=O)=O)CCC(C2CC2)(NC(=O)CN2CCN(CC)C2=O)C1 n1(CC)nc(C(N2CC(N(C(=O)CSc3nc[nH]n3)C)C(F)C2)=O)ccc1=O N1(C(=O)NC2C(C(C)(C)C)C2)CCC2CC(O)CCC2C1 Cc1ccc(Cl)c(C(N2CCC(CN(C(=O)C(c3ccnn3C)C)C)CC2)=O)c1 O=C(O)C1CCCn2nc(CN(Cc3cccnc3)Cc3nccs3)nc21 C1(C(N(CC=C)C)=O)C2CC(O)C(C2)N1C(C1CC2CCCC2C1)=O C1(NC(c2cc(CC)no2)=O)CC(NC(C2(CSC)CC(F)(F)C2)=O)C12CCC2 CC(C(F)(F)C(F)(F)F)=CC(=O)NCCCN1CCN(C(C2CCO2)=O)CC1 C1(C(=O)NCC2(CCOC)CC2)CN(C(c2c[nH]nc2C)=O)CCO1 Cc1ccc(NC(C2CC(F)CN2C(=O)C(=O)C(C)C)=O)c(F)c1F N1(c2c(C#N)cncn2)CCC2(CC1)CC(CO)C2.c12ccccc1S(=O)(=O)N2 CCCC(C)(C)CC(=O)N1CC(NC(=O)C(C2CCC2)C2CCC2)CCC(O)C1 C1(C(=O)NC(CC=C)CNC(c2ccc(SCC)cn2)=O)OCC2CCCC12 CC1=C(C(=O)NC2(C(N(CCC(C)N(C)C)C)=O)CCCCC2)CCC1 C=CCCCC(C(=O)NCC(C1CCCCC1)O)NC(C1CC(=O)N(C)C1)=O N1(C(c2cnc(SC)s2)=O)CCN(C(c2cc(C3(O)COC3)on2)=O)C(CO)C1 C1(O)(C(C)C)CCCN(C(C2(NC(=O)C=CC(F)(F)F)CC(O)C2)=O)C1 C(=O)(CCC=CBr)NCCCN(C(Cc1ccn(CC)n1)=O)C(C)C c1(C(=O)NCC(CO)NC(CNC(C)=O)=O)cc2c(ccn2C)s1 C1(CC(=O)NCC2CN(CP(C)(C)=O)C2)Oc2ccccc2NC1=O C1(C#N)(NC(CCCC#C)=O)CCN(C(=O)Nc2cc(F)ccc2C)C1 C=CC1(C2(C(=O)NC3CN(C(c4c(C)noc4C(F)(F)F)=O)C3)CCC2)CCC1 CCCC(CCC)=CC(=O)NC1CCCN(c2nnc(C(C)(C)C)s2)C1 c1(C(=O)NC2(CO)CCN(C(CCC(C)C)=O)C2)nc2ccccc2[nH]1 c1(C(N2CC(CNC(=O)CN3CSCCSC3)C2)=O)cccc2occc12 C1(NC(C(CCC)OC)=O)CC2(C1)CC(NC(=O)CC(F)(F)F)C2 c1(-c2cn(C(C(=O)NCC3CN(S(CC)(=O)=O)C3)C)nn2)ccn(C)c(=O)c1 c1cc2c(N3CCC(c4n[nH]cc4-c4nn[nH]n4)CC3)[nH]nc2cn1 N1(C(c2ccc(C)n2C)=O)CC2(CCCC2NC(=O)CSC(C)(C)C)C1 C(CCCCCC(=O)NC(c1ccccn1)CO)NC(c1ccc(SC)o1)=O c1(C(=O)NCC(CC(C)C)NC(=O)CC2CC23CC3)cccc(C(F)(F)F)c1F C(=O)(C(C)(C)CCS(C)(=O)=O)NC1C(NC(CCCCCC(C)=O)=O)CCOC1 c1(OC)ccc(C=CC(=O)NC2CCC(NC(C3(C)CCC3)=O)CC2)cc1O CN(CC(=O)c1cccnc1)N1CCN(C(C2C3CCCC23)=O)CC1 N(C(=NCCCF)NCC1CCCS1)Cc1ccc(O)cc1 C(=O)(C(F)(F)CCCNC(=O)OC(C)(C)C)NCc1c(COC)cccc1 C1(C(N2C(C)(C)C(NC(=O)CCCn3ccnc3)CC2)=O)CCCCC12CCC2 n1(C(c2onc(C3N(C(C4CC(C)(SC)C4)=O)CCCC3)n2)=O)ncc(O)nc1=O c1(C2C(C(=O)NC3CC(NC(C4COCCO4)=O)C3)C2)ccc(Br)s1 c1(CC(=O)NCC(CC)NC(c2ccc[n+]([O-])c2)=O)nccc2ccccc12 CC(=NO)C1CC(C(=O)NCC2CCCN2C(=O)C=C2CCSCC2)C1(C)C C1(OC)(CNC(c2ccnc(C3CC3)c2)=O)CCN(C(c2cnc(Cl)s2)=O)C1 C1(CNC(=O)CC2(O)CCC2)CC2(CCN(C(c3csc([N+](=O)[O-])c3)=O)C2)CO1 C(=O)(CS(=O)(=O)N1CCN(C2COCC2NC(=O)C(N)=O)CC1)OC C12(C(=O)NCc3c(CN(C(=O)CCS(C)=O)C)cccc3)CCCN(CC1)C2 N1(C(c2cc(Br)ccc2C)C(=O)NCCOC)CCC(F)(F)CC1C C#CCC(CC(=O)NCCCCCCC)NC(c1cc(OC)nn1C)=O C(=O)(C#CC1CCCO1)N1CC(O)CC(NC(c2ccnnc2O)=O)C1 Cc1nc(O)ccc1C(=O)NC(C1CC=CCC1)C(=O)NCc1ccc(CO)s1 c1(C(=O)NCCCOCCC(=O)NC(C2CCCC2)C#C)ccc(C)c(C)n1 C1(C)(C(=O)NCC(C)(C(C)C)NC(CCc2c(C)nccc2)=O)CCC(=O)NC1 C1(CC(=O)NC2CC(CNC(C3NC(=O)OC3)=O)C2)CCCC(F)(F)C1 C1(CN(C(c2nocc2Cl)=O)C2CC2)CCCCN1C(=O)COCC1CC1 CC1(C)CCC(CC(=O)NC2CCCC(NC(C3(C#N)CCCOC3)=O)C2)CC1 c1(C(N)=O)n[nH]c(=NCCC2CCCN(C(=O)Cc3cc(F)nc(F)c3)C2)s1 C1(NC(c2c(C)nns2)=O)CCCN(C(=O)CCC2CCCN2C)C1 C=CCC(C)C(=O)NCC1CC(O)CN1C(=O)CSCc1ccc(Cl)s1 C1(=O)C(C)C(C)NC(=O)CCOC(=O)NCCO1.C(CC(C)C)=CC.C(C)(C)(C)O c1(N(CC(CN(C(c2c(C)noc2C)=O)C)O)C)cc(Cl)nc(C(F)(F)F)n1 c1(C(=O)NCCN(C(C(CCC)O)=O)C(C)C)ccc(OC(F)(F)F)cc1Br CC(C)(C)CC(O)CC(=O)NC1CC(C)(NC(=O)COCc2nccs2)C1 C12(NC(c3ccc(C)s3)=O)CCC(CN(C(c3csc(C)c3C)=O)C1)C2 CC1OC2(C)CC1(C(N1CCOC(CNC(C3C4CCCC34)=O)C1)=O)C2 Cc1nn(CC2CC2)c(C)c1NC(=O)C(C)NC(=O)NCCOCC(N)=O N12CC3CCN(CC13)C(=O)C1CC1CNCCC2=O.CCCCCN(CC)CC c1(C(=O)NC2C(NC(c3c(C)nsc3)=O)CC2)cccc(-c2nnco2)c1 C(C(C(=O)NCC1CC1[N+](=O)[O-])NC(=O)CCOCC1CC1)N(C)C C1(C(=O)NC2CN(C(COCC(=O)NC)=O)C(C)(C)C2)Cc2ccncc2C1 C12(C(=O)NCc3c(CC)nns3)CCCC1CN(C(=O)C(C)(C)C#N)C2 c1(NC(C2C(C(=O)OC)C2)=O)cc(Br)ccc1C(=O)Nc1ccc(Cl)cc1O C1(F)(CNC(C2(CC(C)C)CC2)=O)COCCN(C(C2COC(=O)C2)=O)C1 c1(C(=O)NCCc2nccs2)cncc(-c2ccc(OCC(F)F)cc2)n1 C123CC(CO)(C1)OC21CN(C1)C(=O)OC3=O.c1(C(C)C)nnc(SC(C)(C)C)o1 C1(CNC(=O)CC2COCCO2)CC2CCC1N(C(c1ncnc(O)c1Cl)=O)C2 C1(NC(CCSCCOC)=O)CC(NC(C2(O)CC2)=O)CC1O.c1(CO)ccncc1 c12ccc(c(Br)c1)C(C)NC2.c1(CC)c(C)noc1C Cc1ccc(NC2CC(=O)c3ccccc32)c2[nH]ncc12 Cc1nn(C)c(C)c1CC(=O)NCC1(C)CCC(NC(=O)C(O)C2CCC2)CC1 Cc1ccc(C=CC(=O)NC2(C)CC(NC(=O)CC3CCC(=O)C3C)C2)o1 c1(C(=O)NC(C2CCN(C(C3CCCC3O)=O)CC2)C)snc2ccccc12 C(C1=NOC2(CCC2)C1)NC(C1CCN(C(CC2(CC)CCC2)=O)CC1C)=O c1(CNC(C2CCN2C(=O)C(c2ccc(Cl)cc2)O)=O)c(F)ccc(F)c1F Cc1c(CNC(c2c[nH]nc2CCNC(=O)CS(C)(=O)=O)=O)cnn1C c1(CC(=O)NC2(CO)CCN(C(=O)CC3CCCO3)CC2)c(F)cccc1Cl C1(CNC(CCC)CC)CCC(F)(CC(=O)OC(C)(C)C)C1 C1(CC)CCN(C(=O)CN(C(C2CC(=O)OC2(C)C)=O)C2CC2)CCO1 C1(CNC(C(CC#C)C)=O)COCCN(C(=O)Cc2cc(C(F)(F)F)c(O)nn2)C1 c1(NCC2N(C(=O)C=CI)CCC2)ccnc2ncnn12 N1(C(COC2(C)CCC2)=O)CCC(CCNC(C2OCC2(C)C)=O)CC1 C1(CC(N)=O)CCC2CNCCC2C1.N1(C(C)C)CCCC1CNCCS(=O)(=O)O C1(C(=O)NCC2(CNC(c3ccc(C#C)o3)=O)CCOCC2)CC(=O)NC1(C)C N1(C(=O)CNCc2cc[nH]n2)CCC(N2CCC(O)C2)CC1 N1(CC(=O)NC2CCC(NC(C3(CC)CC3)=O)C2)CCC(=O)NC1=O C(=O)(C1=CS(=O)(=O)CCC1)NCC1(CNC(C2C(C)C2)=O)CCC1 C1(CNC(CC(C)(C)OC)=O)CN(C(c2ccc(C)nc2O)=O)C2CCN1C2 c1(CC(N2CC(NC(CC(=C)C)=O)C3C2C3)=O)ccc2cc[nH]c2c1 C1(CSC)CCC(NC(C2(C)CC2)=O)C1.c1(C2C(=O)N2)ccccc1.C(C)(C)S CCC(C)C(O)C(=O)NCC12CC(NC(=O)CC(F)(F)Br)(C1)C2 C1(C(=O)NCCCN(C(=O)Cc2ccoc2)C)CC(c2cccc(Cl)c2F)=NO1 C1(C)(CNC(C2(CCCC)CC2)=O)CC(OC)CN1C(C1CC(C#N)C1)=O c1(C(=O)NC2(C)CCCN(C(CNC(CC)=O)=O)C2)ccc(S(=O)(=O)CC)cc1 c1(C(=O)NC)cccc(NC(C2(C)CCN(c3ncc(C(C)C)cn3)C2)=O)c1 C1(C(=O)NC2CCN(C3CC3)C2)(CNC(=O)CCOCC(F)(F)F)CC12CCC2 c1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)O3)=O)C2)cc2ccccc2cn1 Cc1cccn2cc(C(N3CCC(CNC(=O)C4CC4)C3C3CC3)=O)nc12 Cc1cc(C(=O)N(C2CC2)CC2CCCN2C(c2ccc(CO)o2)=O)nc(C)n1 c1(C(N2C(CC(=O)NCCCC3(O)CCC3)COCC2)=O)occ2c1CCC2 Cn1cc(C(N2CC3CC(C2)C3NC(c2ccc(F)cc2O)=O)=O)ncc1=O c1(-c2c(C(=O)NC(C)CN(C)C(C3CSCCS3)=O)c[nH]n2)cc(F)cc(F)c1 Cc1c(-c2cnc(CNC(c3ncn(C)c3Br)=O)nc2)cccc1F N1(C(C2N(CC)CC2)=O)CC(CNC(=O)CC2CCC(C)(C)O2)C(C)C1 CCC(C)C(O)C(=O)NCc1nnn(C)c1C(=O)N.C1(C(=O)OC)(CF)CCCC1 c12cnc(nc1)CNC2=O.c1(CCC(=O)N(C2C(C)CC2)C)cccnc1.C(C)(=O)O c1(C(=O)NC2CCC(CNC(C3C(C)CCS3)=O)CC2)ccc2cccnn12 CS(=O)c1cccc(C(N2CCCC3(NC(c4ccon4)=O)CC3C2)=O)c1 C1(CC)CCN(C(=O)CC(C)SC2CC2)C(C(=O)NC2CC(CCF)C2)C1 C1(CNC(c2ccn(CC)c2C)=O)CN(C(=O)CNC(=O)C(C)(C)C)CCC1C c1(CNC(CCCCC#C)=O)nnc2n1CCN(C(=O)C(O)CCCC)C2 C1(N(C)C)CCCC1NC(=O)COC1CCN(C(=O)Cc2cnc[nH]2)C1 c1(C(=O)NCCCCN(C)C(C2CCCCC2(C)C)=O)c(F)ccc(O)c1F N1(C(C(CC)N(C)CC)=O)CCN(C(c2ccn(CC)c(=O)c2)=O)CC1CO c1(C(=O)NCCC2CCCN(C(C(C)CN(C)C)=O)C2)cn(C)c(=O)n(C)c1=O N1(C(COCCCCC)=O)CC2CCC1CC2NC(c1cnncc1O)=O C#Cc1cn(C)nc1C(=O)N(C1CCCC(NC(c2cncs2)=O)C1)C CC(C)(C)C(O)C(=O)NCC1C2CN(C(c3ncc(Cl)cc3O)=O)CC12 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(C)NC(c2ccccc2F)=O)OCC1 N1(C(CN(CCC=C)C)=O)CCOCCCC1C C1(NC(c2nnc(CC)s2)=O)CCCN(C(=O)CCc2cc(C)[nH]n2)CC1 C1(NC(CC(CNC(c2cn(CC)nc2C)=O)C)=O)CCOCC1(C)C c1(CCC)nc(C)c(C(N2CCCC2C(C)NC(c2ccnn2CCC)=O)=O)s1 c1(COC)nocc1CN(C)C.C12CC1(C)NS(=O)(=O)C2 C1(CNC(CCN(C(C2(c3cccnc3)CC2)=O)CC)=O)CC(C#N)C1 C1(NC(Cc2c(C)occ2)=O)CCCCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(Cc2n[nH]c(=NC)s2)=O)C2CCCC1CN(C(c1conc1C)=O)C2 c1(C(=O)NCC(CN(C(c2cc(C)[nH]n2)=O)C)(C)C)ccc2c(n1)CCC(C)C2 c1(C(=O)Nc2ccc(O)nc2)cnc2ccncc2c1 c1(CC)ncccc1C(=O)NC1CCCC1C(=O)NC(C(F)(F)F)C1CC1 c1(N(C(=O)CC2CC2CNC(=O)COC2CCOCC2)C)cccc(C(N)=O)c1 N1(C(c2ccc(CC)o2)=O)CCC(O)(C(C)CNC(c2ccsc2Cl)=O)C1 C1(C2CCN(C(=O)C(O)C3CCC3)CC2)(NC(=O)CNc2ccccc2Cl)CC1 C=CCC(CC(F)F)NC(=O)C1=NOC(CNC(=O)COC2CC=CC2)C1 C=CCC(C(=O)N1CC(NC(c2ccc(OC)cc2C)=O)C1)C(C)(C)C c1(C(N2CC(N(C(=O)CNS(C)(=O)=O)C)C2)=O)ccccc1 N1(C(Cc2n(C)ccn2)=O)CCC2CN(C(=O)CC3CCCS3(=O)=O)CC2CC1 c1(C(N2C(CNC(C)=O)C=CC2)=O)cccc(N2C(=O)CCC2=O)c1 C1CCCCC(=O)N1.C1(NC(C(CCC)N(C)C)=O)CC2(CCCO2)CC1 Cc1nc(C2CC2)ccc1C(N1CCOCC1CNC(=O)CC1CCC2CC12)=O c1(C(N2CCCC2C2(C(N3CC4(CNC(=O)N4)C3)=O)CC2)=O)c[nH]c2nccc-2c1 CC1(C(N2CCC(NC(=O)CC3CCOCC3)C2)=O)CNC(=O)C1 c1(NC(c2ccoc2)C)nccc(NC(CCO)c2nccs2)n1 C1(NC(c2n[nH]c(C)c2O)=O)C2CC1CN(C(=O)Cc1cc(F)ccc1Br)C2 C1(C(=O)N(C2CCN(C(c3c[nH]nc3C)=O)C2)C)(OC)CS(=O)(=O)C1 c1(NC(C2(O)CN(C(=O)CC3COCC(C)(C)O3)C2)C)ncnc2c1ncn2C CN1CCCC(C(=O)N(CCC(=O)NCCCS(N)(=O)=O)CCCO)C1 c1(OC)ccccc1C(=O)NC1CCC(N(C)C(c2cc(OC)ccn2)=O)CC1 Cc1cccc(C(=O)NC2CN(C(=O)C(C(C)C)N3CCCC3=O)CC2O)c1Cl C(CN=c1[nH]c(=N)[nH]c(=NCC(C)c2ccc(Cl)cc2Cl)[nH]1)N(C(=O)OCC)C Cn1cc(C(=O)NCCN(C(C2C=CC=CC=C2)=O)C2CC2)c(-c2ccco2)n1 C1(C(=O)NC2(C)CCCN(C(=O)COCCF)C2)OCC2CCCC1C2 c1(C(=O)NCC(CNC(c2cc(C)nn2C)=O)O)nc(O)c2ccccc2c1C CC1(C)CCCN(c2ncccc2SC2CC2)C1CCO C1(C(=O)NCCNC(=O)Cn2cc3ccccc3n2)CN2CC3CC2(CO1)C3 CCC#CCN=c1nc(N2CCC(c3ccc(CO)o3)CC2)c2ccccc2[nH]1 Cc1cc(CNC2CC3(C2)CC(NCc2cccnc2)C3)cc(O)n1 N1(C2C(=O)N(CCCF)C(=O)N2Cc2ccccc2)CCCC2(COCCO2)C1 Cn1cc(CC(N2CCC2(C)CC(=O)NC2(C(N)=O)CCOC2)=O)cn1 N1(C(CCNC(Cc2c(C)n[nH]c2C)=O)=O)CC2CCCCC2C1 S(=O)(=O)(c1ccc2c(c1)CCO2)N1C2CCN(C(=O)CCSc3cccs3)C2CC1 CN1CCc2cc(C(=O)NC3CC3NC(C3(C)CCCNC3=O)=O)ccc21 N1(C(C(C(C)OC)OC)=O)CCCc2cnnc(O)c21 N1(C(c2csc(C)c2C)=O)CCCC2C(NC(=O)CCC(C)(C)F)C(C)(C)C12 CC1(C)CC1(C)C(=O)NCC1(CNC(c2cc(Br)n[nH]2)=O)CCC1 c1(CC(=O)NC2CN3CCC2O3)ccc(S(=O)(=O)NCc2ccc(CO)cc2)s1 N1(C(c2cc(CC)oc2C)=O)CCC(C(=O)NOC(C)CC)CC1(C)C C(C(=O)NC1CC(C(N)=O)C1)(C(F)(F)F)OC(C)=O.c12cnc(s1)C(C)NC2=O c1(C(=O)NCC=CCNC(c2c(CC)occ2)=O)nccc(Br)c1C Cc1nn(C)c(C)c1COC(=O)C(O)Cn1cncn1 c1(CC(=O)NCC2CN(C(c3c(C)cc(C)[nH]3)=O)CC2O)c(Cl)cccc1Cl Nc1nc(Cl)ccc1C(N1CC2CC1C2NC(c1ccc(Br)o1)=O)=O Cc1ccc(C(=O)N(C2CCCCN(c3cc(C(N)=O)ncn3)C2)C)nc1O C1(C(=O)NC2(CCOC)CCCC2)CC(C)(C)CN1C(C1CC1C(C)C)=O CC1CN(C(=O)CC2CCCC2NC(c2ccncn2)=O)CC(C)(C)O1 c1(C(=O)NC(C2(O)CN(C(C(C)c3cc[nH]n3)=O)C2)C)cn2c(n1)COCC2 N1(C(C)=O)CCCC1C(=O)NC1CCC(CNC(=O)C(C)CN(C)C)C1 C1(C(=O)NC(CC)C)CN(C(c2cc(F)c(F)cc2I)=O)CCC1(F)F C(=O)(C1CCCc2sccc21)NCCN1CCN(C(C2C(C)C2C)=O)CC1 Cc1cc2c[nH]nc2cc1C(=O)NC(C)(CNC(c1cnn2ccsc12)=O)CO CCCC(O)(CNC(C(C)(F)F)c1ccccc1)C(F)(F)F CC(C)C(F)C(=O)N1CCC(NC(=O)C(c2ccc(F)cn2)(F)F)C1C n1(CC)nc(C(=O)NC2CCCCC2CC(=O)NCc2cc(C)cs2)cc1O C1(NC(c2ncc(OCC)nc2)=O)CCN(C(=O)C=CBr)C(c2ccccc2)C1 C1(C(=O)NC(C)CN(c2cc(Cl)nc(C3(C)CC3)n2)C)CNC(=O)CC1C N1(C(C(N2CC(C)(CNC(CCNC(=O)NC)=O)C2)=O)C)CCCCC1=O C(=O)(CC(C)C(F)(F)F)NCCC1CC(OC)CN1C(c1cnn(C)n1)=O CC(CC(F)(F)F)C(=O)N1CC(CNC(c2ccc(CO)c(Cl)c2)=O)CC1(C)C Cc1c(C(=O)NC23CCC(C2)N(C(=O)CC2CCC2)C3)c(C(F)F)nn1C Cc1nc(Cl)ccc1CC(N1CCC(C(C)NC(C2CC(C)CO2)=O)CC1)=O c1(CCC)cc(C(=O)N(C)Cc2csc(COC(C3CN(C4CC4)C3)=O)n2)nn1C N1(C(c2c(CC)cco2)=O)CCC2(CC1)CC2NC(=O)CN1CC=CC1 C12CCN(CC1CO)C2=O.c1(NC(=O)C=CC2CCOC2)c(CO)cccc1F N1(C(=O)CC2CCOC2)CCCC(C2CN(CCN3CCCC3=O)C2)C1 c1(CNC(=O)NC(C2CCOCC2)C)ccc(C(=O)N(C)C)cc1.C1CCN1 C(=O)(C1=CC(O)C(C(=O)N(C)C)C1)NCCOCCNC(C)C c1(C(C(=O)N(C(C(CC)O)C)CCC#N)(C)C)ccc(Br)c(C)c1.OCC C=CC1CCC1C(=O)NCCOCCNC(C1(CF)CC1(F)F)=O c1(OC)ccc([N+](=O)[O-])c(C(N2CCC(NC(c3cnns3)=O)C(CO)C2)=O)c1 C12(NC(c3cn4cc(C)nc4s3)=O)CCOCC1CN(C(C1(C(F)F)CC1)=O)C2 C(=O)(CC(C)CC(C)C(CC(C)=O)OC)N(c1cccc(C)c1)CC C1(NC(C2(F)CCC2)=O)(COC)CCN(C(CC2(C(=O)OC)CC2)=O)CC1 CCCCCC(CC)C(=O)N1CCCC(F)(CNC(C2C3CCCC23)=O)CC1 C12(CNC(C3C(C)C3)=O)CCCCC1N(C(c1ccc(F)c(O)c1F)=O)CCC2 C#CCCCC(C)C(=O)N(CC(=O)NC(C)CC(C)(C)OC)C1CC1 C1(C(N2C(C)COCC2)=O)CCN(C(=O)C2CCC2C)O1 c1(CNC(C(C)C)=O)nnc2n1CCN(C(=O)Cc1ccc(Br)cc1)C2 c1(C(=O)NCCC2CCC(NC(COCC)=O)C2)ccncc1Br c1(NC(C2CN(Cc3cc(B(O)O)co3)CCN2)=O)nc2cc(Cl)ccc2s1 C=CC(C)(O)CC(=O)N1CCC(NC(c2cc(Cl)ccc2OC(F)(F)F)=O)CC1 Cc1cc(-c2cn(CCC(=O)NCC3OC(=O)NC3(C)C)nn2)cc(C)n1 C12(CC)CCC(C(N3CCC(CNC(c4ccncc4F)=O)(OC)C3)=O)(CO1)C2 C#Cc1ccc(C(C(=O)NCCCC2CC2)N(C)Cc2n[nH]cc2CC)cc1 C(=O)(C(F)(F)C(F)(F)F)N1CC(C)(NC(=O)CCc2ccc(F)nc2)C1 C(=O)(C(C(C1CC1)OC)N(C)CCN1CCCCCC1)NCCC(=O)OCC c1(OCCC(=O)OC)ccccc1CN1CCN(c2nncn2C)CC1 C1(C(=O)NC(CC(C)C)CO)CC2(CC2)CN1C(c1ccc(I)cc1F)=O C(=O)(C(F)CCC(C)C)NC1C(NCC(=O)N(c2cc(C)cc(C)c2)C)CCC1 C1(CC(=O)NC(C)CC2CN(C(=O)CNC(=O)CN(C)C)C2)CCCCCC1 C1(C(=O)NC(CC)CNC(c2cc(C)c(C)o2)=O)CCCN(S(N)(=O)=O)C1 CC1(CCNC(C2CCC(=O)NC2)=O)CCN(C(C2(C)COC(=O)C2)=O)CC1 N1(C(C=CCC)=O)CCCCCC1CNC(c1c(Cl)cncc1Br)=O C1(NC(C)=O)COCCC1NC(c1ccc(-c2ccccn2)nc1)=O C1(NC(CNCc2ccc(C)s2)=O)CCOCC1NC(=O)Cc1cncnc1O C1(C(C)NC(CN(C)CC)=O)CCN(C(=O)CCCOC(C)=O)C1.C(C)(C)(C)O C#Cc1cccc(C(=O)NCCCCNC(C2CC3(C)CC2CO3)=O)c1 N1(C(C=CC)=O)CCN(C(c2csc(COC)n2)=O)C(CC)C1 Cc1cnc(Cl)cc1NC(C1(C)CCN(Cc2ccc(F)c(O)c2)CC1)=O CC(CC(C)(C)O)N1CCC(CNC(C2(c3ccc(F)cc3)CCCC2)=O)C1 C(CCCC(=O)N1CCC(O)C1C(C)(C)C)N(C(C(SC)SC)=O)C C=CCCCCN=c1nc2ncn(C)c2c(NCC2CCCN2CC(F)F)[nH]1 Cc1cc(C(=O)NC2(CNC(=O)CNC(=O)CC(F)(F)F)CC2)nc(O)n1 c1(C(=O)NCC2(NC(C(CCOC)C)=O)CCC2)ccc2[nH]c(=N)oc2c1 N1(C(C2CCCC(C)CC2)=O)CCCN(C(c2ncnc(O)c2F)=O)CCC1 C(=O)(C1=CCCCCC1)NCC1N(C(C2CC(C)OC(C)C2)=O)CCC1 N1(C(C2C(CNC(C(C(C)C)OC)=O)CCC2)=O)CCC2(CC1)CN(C)C2 C=CC(CCC)CC(=O)N1CCOC(CCNC(c2ccc3c(c2)COC3)=O)C1 c1(C(=O)NC2CC3CN(C(C(CC)C)=O)CC(C2)C3)cnc(O)c([N+](=O)[O-])c1 CC(F)CN=c1nc2c(cnn2C)c(N(C)Cc2ccc(Br)cn2)[nH]1 C1(CC)CN(C)CCCN1C(C1CC(O)CN1C(=O)C(Cl)Cl)=O C=CC1CCN(C(=O)NCCNc2cnn(-c3ccccc3)n2)C1 CCC(CNC(=O)C(F)(F)c1ccsc1Cl)(CC)NC(=O)CCN(CCO)CCO C1(C(=O)OCC)CCC(n2nc(C(C)(C)SC)nc2-c2ccncc2O)CC1 C1(C(=O)NCC(C)NC(C2CC(OC)C2)=O)CC12CCOc1ccc(F)cc12 C1(NC(=O)OC(C)(C)C)Cc2nn[nH]c2C(C)C1.CCCC(CCC(=O)OCC)N c1(CC2(NC(c3cc(C(=O)NCC4(OC)CC4)on3)=O)CC2)cc(C)ccc1C C=CCC(CC(C)C)C(=O)NCC1(C(N)=O)CN(C(=O)CN2CCCCC2=O)C1 CC(C)(C)C#CCCNC(C1COCCN(C(=O)C=CC(F)F)C1)=O N1(C(CC2(C)CCCCC2)=O)C2CCC1CC(CNC(=O)C=CC1CCOC1)C2 c1(C(N(C(C(=O)NCC2CCN(C(C)C)CC2)(C)C2CC2)C)=O)cc(O)ccc1F C12(NC(c3cc(F)ccc3F)=O)CCC(C1)N(C(=O)CCOC1CCCC1)C2 Cc1cccc2cc(C(=O)Nc3cccc(-c4nc(O)n[nH]4)c3)[nH]c12 c1(C(=O)NC2CC(C)N(C(c3csc(=N)[nH]3)=O)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC(C)O)c[nH]c2ccc(-c3cccc(NCCF)c3)cc12 n1(CC)nc(C)c([N+](=O)[O-])c1NC1CC(NC(=O)Cn2cnc3c2CCCC3)C1 c1(C(=O)NC23C(CN(C(CS(CC)(=O)=O)=O)C2)C3)cc(F)c(C#N)c(F)c1 C1(C(=O)NC2CCCC2O)(CNC(c2cc(Cl)cs2)=O)CCCC1 C(=O)(C=C1SCC(=O)N1C)N1CCCC(CCC)(NC(c2nc(Cl)oc2C)=O)C1 CC(C(=O)NCC1CN(C(=O)C(C)(C)n2cccn2)C1)C(F)(F)F c1(OC)c(CN2CCN(C)CC2)cc(Cl)cc1-c1cc[nH]n1 c1(C(=O)NCC2N(C(c3cc(C)n(C)n3)=O)CC2)coc2c1CSC2 N1(C(=O)NC2C(c3n(C)ccn3)OCC2)CCCC2CCC12 c1(C(=O)Nc2cccc(CN(C(C)C(N)=O)C(C)C)c2)cc2c(ccn2C)[nH]1 C1(C)(CNC(C=COCC)=O)COCCN(C(c2c(C)noc2N)=O)C1 C(CC(F)(F)F)NC(c1cn(CC2CCCO2)nn1)=O c1(OC)cncc(C(=O)N(C(C)C(=O)NCc2csc(C)c2C)C2CC2)n1 c1(OCC(=O)NCC2CC(NC(c3c(C)nsc3)=O)C2)cccc(Cl)c1 C1(NC(c2cc(C)nnc2O)=O)CCCCN(C(=O)C(C)(Cl)Cl)CC1 N1(C(CC2CCCN(C(C(C)CC3CCC3)=O)CC2)=O)CC2(CCCCC2)C1 C1(C(N2CC(C(N)=O)(CNC(C3(C)CCCCC3)=O)C2)=O)Cc2ccccc2O1 C1(NC(C2CCCN2C(=O)C2CC2)=O)CCOC12CCN(C(=O)CCC(F)F)CC2 c1(C(=O)NCCCc2ccc(C)nc2)cc(C)nc(-c2ccccn2)n1 c1(C(=O)NCC(CNC(C2CC2c2cccs2)=O)OC)cc(O)cc(Cl)c1 CCCCC(CNC(c1nncs1)=O)NC(=O)C(C)Cc1ccc(N)cc1 n1(CC)nc(C(=O)NC(CNC(=O)CCSc2ccccc2)CO)c(C)n1 C(=O)(C(C1=CCCSC1)N1CCCC(c2ccccc2)(COC)C1)NCC(=C)C CCCC(CNC(=O)CCOCC)NC(c1cc(=N)[nH][nH]1)=O CCC(CC(=O)N1CC(CC(C)NC(c2sccc2S(N)(=O)=O)=O)C1)C(F)F c1(NC(C)=O)ccc(N)c(C(N2CC(N(C)C(C3CCCO3)=O)C(C)(C)C2)=O)c1 c12sccc1C(=O)N2.C1(C(C(C2CC(NC(=O)OC(C)(C)C)C2)C)=O)CCCO1 C(C(C(=O)N1CCCC1CCCNC(c1cn(CCO)nn1)=O)NC(C)=O)OC N1(C(C2C(C(=O)NCC#C)C2)=O)CC2(CCC2)CC1CNC(=O)CC(C)N(C)C C1(NC(C(=Cc2c(Cl)cccc2Cl)C)=O)CCC2CN(C(=O)CNC=O)CC2C1 CC1(C)CN(C(=O)C(c2ccoc2)NC(c2nccs2)=O)C2CCCC12 Cc1cc(F)cnc1C(=O)NCC1CC2(CC2)CN1C(=O)CN1CCNC(=O)C1 c1(SCC(N2CCC(O)(CNC(C3(C=C)CC3)=O)C2)=O)ccc(C#N)cc1 C1(N(C(=O)Cn2cc(CO)nn2)C)CCC(NC(c2cnc(OC)nc2)=O)CC1 c1(C(=O)NCC(C)(C)CCNC(c2cccnn2)=O)scc2c1CCCC2 CC1(C)CC(CC(N2CC(CF)(NC(=O)C(Cl)=CCl)C2)=O)CO1 C(=O)(C1CCCn2cncc21)NCC(COC)NC(c1nsnc1O)=O C1(C(=O)NCC(C)NC(c2cc(C)no2)=O)CCCCC12CCC2 N1(CCN(C(C2(CC)CCCO2)=O)C)CCN(C(=O)CCc2ccccc2)CC1 N1(C(C)C(=O)NC2CCCC2)CCCC12CCN(C(=O)NC1CCCSC1)CC2 C1(NC(c2c(CNC(C(CN(C)C)(C)C)=O)ocn2)=O)CCCC(F)(F)C1 C1(CNC(=O)C=CCF)CCC2(CCC2)C1NC(=O)COc1ccccc1[N+](=O)[O-] Cc1cc(N2Cc3c[nH]nc3C2)nc(N2CCCC(CO)C2)n1 Cc1ccc(Cl)c(OCC(=O)NCC2(F)CC(NC(=O)C(=O)N(C)C)C2)c1 C12(CNC(C(C=CCCC)O)=O)CC1CN(C(c1cnn(CC)c1Cl)=O)C2 C1(C(=O)NC2CC(OC3CC3)C2)CC(O)CN1C(=O)CCc1ccncc1 c1(Sc2n(C(C)Cc3ccccc3)c(-c3ccco3)nn2)cccc(C#N)c1 c1(C(N(C)CC2(NC(C3CC4CCC3O4)=O)CC2)=O)cc(=O)n(C)o1 C1(C)(CC)CC(NC(c2ccnnc2)=O)CN1C(c1cccc(Cl)c1OC)=O CC1C(NC(C2CC2(F)F)=O)CCCN1C(C1(C)CCCC1C)=O Cn1ncc(CNC(C2(C)C=CCCC2)=O)c1C(=O)NCC(c1cccnc1)O C(=O)(CCCCC(F)(F)F)N1CCN(CCNC(c2c(CC)cncc2)=O)CC1 Cc1cc(Cl)ccc1-n1nc(CCC(C)C)nc1C1CCCN1CC(C)C c1(C(=O)NC2CCN(C(c3ccc(COC)o3)=O)C2)ccc2cnccc2n1 c1(C(N2CCC(OC)(CNC(c3ncccc3C)=O)C2)=O)ncc(C)cc1C CC(C)C(O)CC(=O)N(CCNC(c1csc(NC(N)=O)n1)=O)C(C)C N1(C(C)=O)CCc2cc(CNC3(c4nnnn4C)CCOCC3C)ccc2C1 c1(C(=O)NC(C(=O)OCCC)C)ccnc(CNC(=O)CN2CCCCC2)c1 N1(C(C2Cn3c(C)nnc3C2)=O)CCCn2nncc2C1 c1(C(=O)NCCN(CCCC[Si](C)(C)C)CCC)ccc2c(n1)CCO2 Cc1cccc(C(CNC(c2c(C)n[nH]c2C)=O)NC(C2(C)C=CCCC2)=O)c1 C(C)(CNC(c1cc(C)n(C(C)C)c1)=O)(CC(C)C)NC(c1c(OC)ccs1)=O CCS(=O)CC(=O)NCCC1CC(NC(=O)CN2CCC(O)CC2)C1 CN1CN(C(C2COCCN2C(=O)CCCn2ccnc2)=O)CC1=O N1(C(c2cnc(OC)s2)=O)CC2CCC2(CCNC(C2(O)CC(C)(C)C2)=O)C1 C=CCCCC(=O)NC1(C)CN(C(C2(c3ccccc3)CC(F)C2)=O)C1 N1(C(c2cccc(OC)c2)=O)CC=C(C(=O)NC2CCCCC23CC3)C1 N1(C(C2C(C)=C2)=O)CCC(CF)(NC(c2ccc(C3CCOC3)s2)=O)C1 C1(F)(CNC(C(C)SCC)=O)CCN(C(c2cc(C3CCCCC3)n(C)n2)=O)C1 C(C)(C(O)C(=O)NCCCN(C)C(c1cccc(-n2ccnc2O)c1)=O)OC C(=O)(C(CC(F)F)C1CCC1)N1CCN(C(c2cc(C)sc2C)=O)CC1 c1(C(=O)NC2CN(C(C(CCCC)NC(N)=O)=O)C2)nccc2ncccc12 CC1CC(NC(c2cc(N)ccn2)=O)CN(C(C2(CF)CCC2)=O)C1 c1(OCC(=O)NC2C(NC(CC(CC)SC)=O)C2)c(F)cccc1F N12CCC(O)C(C1)N(C)C2=O.C1(CCNC(=O)NC(C)(C)C)CC2CCC1O2 Cc1ccc(C(=O)NC2(C)CC(NC(c3c(C4CC4)cccc3F)=O)C2)cc1F Cc1ccc(F)cc1C(N1CCCC1C(C)(C)C(=O)NC1(C)CSC1)=O c1(C(C)C)ccc(C(N2CC(F)(CNC(C3CCC3C)=O)C2)=O)c(F)c1 N1(C(c2n(C=C)nnc2)=O)CCC(C)C(CNC(=O)C(=O)NC2CC2)C1 c1(NC(=O)NCCn2c(C)ncc2)ccc(NC2COCC(C)O2)cc1Cl N1(C(CCOCCOCC)=O)CC(NC(=O)CC2CSCCS2)CC(C)C1 C1(NC(C(C2CCN(C(c3csc(F)c3)=O)C2)F)=O)CC2CCC1O2 C1(C(=O)NC(C)CCNC(C2(C)CC=CCO2)=O)CCCCCCC1 C1(C(N(CCC(=O)NC2CCC2(C)C)CC#C)=O)C(C)(C)C1(F)F C(=O)(C(C)CCC(C)(C)C)NC(CNC(c1c(C)cc(OC)nc1)=O)C(C)C N1(C(C2C(CN(C)C)C2)=O)CC2CC1CN2C(=O)C=Cc1cncs1 C1(CNC(c2ccc(OCOC)cc2)=O)CC2(CC2)CN1C(=O)C(C)(F)F c1(OC)ccc(OC)c(C(=O)NC2CC(NC(C3CCCC3)=O)C2)n1 N1(C(c2c(C)cccc2[N+](=O)[O-])=O)CC2CN(C(=O)NC3CC3)CC2C(F)(F)C1 c1(OC)ccc(O)cc1NC(=O)CC1CC(NC(c2[nH]cc(C)c2C)=O)C1 c1(C(=O)NC2CCN(C(c3c(C)[nH]nc3Cl)=O)C2)nccc2cccnc12 C(c1ccccn1)=CC(N1CC(F)(CNC(=O)C=CI)C1)=O C=CC(CCC)CC(=O)N1CCCN(C(C2(O)CC2(C)C)=O)CC1 c1(C(=O)NCCC2CC(C(C)(C)C)C2)csc(COC)c1.C1(=O)C(C2CCC2)N1 C1(NC(C(COC)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCCCCC1(F)F C(C(CN=c1[nH]n(C(C)C)cc1[N+](=O)[O-])C(F)(F)F)NC(c1c(C)ocn1)=O C1(O)(C(C)NC(=O)CS)CCCC1.N1(C(CCCNC(C)=O)=O)CCCCC1 C1(C(=O)NCc2cncs2)CN(C(=O)CC2CCCC3CC23)CCO1 C1(O)(CNC(CCSc2n(C)ccn2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)C1 C1(C)(CC)C=C(C(=O)N2CC=C(C(=O)NCCN(C)CCOC)C2)C1 CC1CN(C(C2CCCC(=O)N2)=O)CC1CC(=O)NCC1(CCO)CC1 C1(C)(NC(C2CC(CNC(c3cn(CCC)nc3)=O)C2)=O)CCC(=O)N(C)C1 c1(CC)nc(N2CCCC2CN(C)C(c2ocnc2C)=O)[nH]c(=N)n1 N1(C(=O)CC2(CO)CC2)CCN(C(=O)C2=CCCSC2)C2COCC12 CC1CCC2(CCN(C(=O)CN(C(=O)CCc3ncccn3)C)C2)C1 C1(CNC(c2ccc(C)nc2O)=O)CN(C(c2cc(C)[nH]n2)=O)C2(CCC2)C1 C1(OCC)CCC(NC(c2noc(C)n2)c2nnnn2C(C)(C)C)CC1 c1(NC(=O)NCC(=O)NC(CC(=O)OC)c2ccccc2)ccc(C)cc1C c1(CNc2ccc(CCNC(Cc3ccc(C)nc3)=O)cc2)cnn(C)c1C#N C(=O)(C(CCC1CCCOC1)N(c1ccc(F)cc1)C)NC(C(=O)OC)C c1(-c2onc(C(C)NC(=O)NCCC3SCCS3)n2)ccc(Br)cc1 C1(NC(c2cc(C)ns2)=O)CC12CCN(C(c1ccc(C#N)n1C)=O)CC2 C=C1CCN(C(C2CSC2)=O)C(C(=O)NCc2[nH]c(C)nc2C)C1 N1(C2CCN(C(C(C)CF)=O)CC2)CCN(C(=O)C(CO)C2CC2)CC1=O c1(CN(C(=O)CSc2nnc(S)s2)CCC)cc2cc(Cl)ccc2o1 N1(C(=O)Cc2ccc(Cl)c3ccccc23)COCC2(COCC3CCCN23)C1 N1(C(=O)OC(C)(C)C)CCCC(O)(CNC(=O)NC2CC2C2CCCCC2)CC1 C(=O)(C(CC)CC(C)C)NC(CCCC(=O)NCc1c(COC)noc1)C c1(C(=O)NCCC2CC(NC(CC(CN(C)C)O)=O)C2)ccn2cc(C)nc2c1 c1(OC(C)C)ccc(CC(=O)NCC2(F)CC(NC(c3ccsn3)=O)C2)cc1 N1(C(COC(C)(C)C)=O)CC2CCC1C1CN(C(=O)C=Cc3ncco3)CC21 CC1(C)CC(CNC(C2CC23CCCC3)=O)N(C(c2ccsc2C#N)=O)C1 c1(CNC(C(COCC)NC(CC=CC=C)=O)=O)ccc(O)cn1 c1(CCC(=O)OCC)ccc(NC(=O)C(=O)NCCc2cccc(I)c2)cc1 Cc1nncc(C(=O)NC(C)C(N2CC(C)C2(C)C)=O)c1C c1(C(=O)NCC2(CCNC(c3ccc[nH]3)=O)CC2)nccc2c(F)cccc12 c1(CC(C(=O)N(C(C(=O)N(C(C)C)C)C)C2CC2)C)ccc(F)c(F)c1 c1(C(=O)NC(C2CCN(C(c3c(CC)occ3C)=O)C2)C)cc(C)ccc1C C1(F)(CNC(C2(OCC)CCSCC2)=O)COCCN(C(c2cncnc2)=O)C1 Cc1cc(O)c(Cl)cc1C(=O)NC(C)CCCCNC(c1ccc(N)cc1O)=O N1(C(CCOCC)=O)CCC(F)(CNC(C2CC(O)(CC)C2)=O)C1 C1(C(=O)NCCCN(C(c2nc3cnccc3s2)=O)CC)CCc2nnnn2C1 CC1(C)CC(NC(C2Cc3ccccc3O2)=O)CN(C(=O)CN2CCCCC2)C1 C1(c2nn[nH]n2)(CC(C2CC2)C2CC2)CCOCC1.C12(CC1)C(=O)NC2 C(=O)(C(C)CC(F)(F)F)N1CCOCC(NC(c2nccc(C)c2)=O)C1 C1(CCC(N2C(C=C)CCC2)=O)CCCCN(C(c2nocc2Cl)=O)C1 c1(OCCO)csc(=NCC2C3CCOCC23)[nH]1 c1(C(=O)NC(C(=O)OC)CSc2nc3c(s2)CCC3)cc2occc2n1C Cc1cc(C(=O)NC(C)CC(=O)NC2CSC2)nn1-c1ccccc1 C(=O)(CCCCCN=[N+]=[N-])N(C(C(N1CC(COC)C1)=O)C)C N1(C(C)(C)C)CC(C2CCCN2C(=O)Cc2nccs2)C(O)C1 C1(C(N(C(C)C(=O)Nc2ccc(Cl)cc2)CCOC)=O)(CN)CC2CC2C1 CCCCN=C(NCCc1ccncc1Cl)N1CCN(CC)C(=O)C1 C1(C(=O)NC(C)(C)CNC(C2(Cc3ccccn3)CC2)=O)CC(=O)N(C2CC2)C1 c1(CNC(CNC(CC(=O)O)c2ccccc2)=O)ccc(Br)cc1F N1(C(Cn2c(C)cnc2)=O)CCCC1(C)CNC(C1(C(C)C)COC1)=O C(=O)(C1=CCCCCC1)NCC(CC)NC(c1cccc(C)c1[N+](=O)[O-])=O CCCC(F)C(=O)N1CC(CC(C)NC(c2cnccn2)=O)C1 C1(NC(c2ccc(C)n2C)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC1(C)C N#Cc1cncc(N2CCCC(CNC(=O)COCCc3cccs3)C2)n1 C1(OC)(CNC(=O)C(O)C(C)C)CCN(C(c2conc2C2CC2)=O)CC1 C1(S(N)(=O)=O)(C(N2CC(N(c3cc(C4CC4)ncn3)C)C2)=O)CCC1 c1(CC(=O)NCC=CCNC(C2CN(C(N(C)C)=O)C2)=O)nnc(O)s1 N1(C(C(C)OCCN(C)C)=O)CCCC(CNC(=O)CC2C=CCCC2)CC1 C#Cc1cnn(C)c1C(=O)NC1CC2C(NC(=O)CN(C(=O)COC)C)C2C1 C1(C(N(C2CCN(C(C(C)OCCN(C)C)=O)CC2)C)=O)Cc2ccccc2S1 C1(CC)CN(C(c2c[nH]c(=NC)s2)=O)CCC1CNC(c1cnn[nH]1)=O N1(C(C2CC(CCC)C2)=O)CCC2(CC1)CC(NC(=O)CCC=CBr)C2 Cc1cc(C(=O)NC2CCC(CNC(=O)CC(C)(C)O)C2)nn1C N#Cc1c(Cl)nsc1N1CCC(CC(N2C3CCC2(CO)CC3)=O)C1 c1(C(=O)NC2CN(C(C(CC=CC)CC)=O)C(C)C2)cc(Br)c([N+](=O)[O-])[nH]1 N1(C(C2(CC=C)CN(C(=O)CC3CCC(C)O3)C2)=O)CCC(CC2CC2)CC1 C=CCCCC(C)NC(=O)C(Cc1ccco1)NC(=O)CCOC1COC1 C(=O)(C1=C(c2c(Br)cccc2Cl)N(C2CC2)C(=O)NC1c1c(Br)c(C)nn1C)CC C1(C(N2CCC(CSC)C2)=O)CC(C(C)C)CCN1C(=O)CCc1cncn1C Cc1cc(C(N2CC3C(NC(C4(Cl)CC45CCOCC5)=O)C3C2)=O)c(O)c(C)n1 C=CC(O)C(=O)NCCOC1CN(C(=O)CCC2CCC(C(=O)NC3CC3)O2)C1 C(=O)(C1=Cc2cc(F)ccc2OC1)NC1CCN(C(C=C2CCN(C)C2)=O)CC1 C1(C(=O)NCC2CCN(C(C3(CC=C)CCOCC3)=O)C2)CCCC2(CCC2)O1 c1(C(=O)NCC2N(C(CC(CC)C3CC3)=O)CCN(C)C2)nc(Cl)c(=O)[nH]c1N C1(OCCC(CC)O)CCC12CN(C(=O)OC(C)(C)C)C2 Cc1nccc(CC2CCOC2NC(=O)NC2CC(OC(C)C)C2(C)C)n1 CS(=O)(=O)CCCC(=O)NCC1(CNC(=O)CC2CC2(Cl)Cl)CC1 N1(C(C=CC)=O)CCOCC1C1CCN(C(=O)Cc2cc(OC)no2)CC1 Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NCCN2CCCC2=O)c(C)s1 C1(CCCC)CN(C(C2CCCN2Cc2cn(Cc3csc(Br)n3)nn2)=O)CCO1 Cc1cc(F)c(C(=O)NC(C2(Cc3ccccc3)CC2)C)c(F)c1 Cc1nc2cc(NC(c3cc(F)ncc3NCc3cn(C)cn3)=O)ccc2o1 Cc1ncc(CC(=O)N(CC(=O)NC2CC3(CC3)C2)C2CC2)s1 C1(C(N2C(C)(CC(=O)N(C)CC3CC(=C)C3)CC2)=O)CCCC(N)C1 c1(N(CCCCCOCC)Cc2ccc(C)o2)ccc(Cl)cc1 N1(C(C(COC)COC)=O)CCC(C)(C)CC1C(=O)NC(C)C(O)C(F)F CC1SCCCC1C(N1CC=CC1(C)C(=O)NC1CC(CO)N(C)C1)=O c1(N(C)Cc2nnnn2C)[nH]c(=NCc2coc(CO)c2)nc2c1ncn2C C(=O)(C(C)(C)C(=O)NCC(c1ccnn1C)O)N1CCC(C(=O)OCC)(CO)C1 C#CC1CCN(C(=O)C(c2ccnn2C)NC(c2scnc2Cl)=O)C1 C(=O)(CC1NC(=O)c2ccccc21)N(C1CCN(C(C(COC)(C)O)=O)C1)C Cc1nc2c(o1)CCCC2CC(=O)Nc1cccc(=NCc2cc(C)on2)[nH]1 C(=O)(CS(=O)(=O)C1CC1)NCCNC(C1(C(C)C)CC1)=O C1(C(N2C(CNC(C3(COC)CC3(F)F)=O)CCC2)=O)CC(C)CCO1 C(CCC(C)NC(=O)Nc1cnc(-c2ccoc2)s1)OCC C1(CNC(c2nc(CC)sc2)c2nnnn2CCCOC)CCCC(F)C1 Cc1nn(C)c(C)c1C(C)C(N1CC2(CC2)CC1CNC(C12CC(C)(C1)C2)=O)=O c1(C(=O)NC(CNC(CCCCCCC)=O)CO)cc2cccc(OC)c2o1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1C2(CCC(NC(CNC(C)=O)=O)CC2)C1 C(N=c1nc(C2(CO)CC2)[nH]s1)C1CCC(CNC(c2cc(F)cc(F)c2)=O)CC1 Cc1ccc(C)c(CN2CC3CC2CN3C(=O)C=Cc2ccc(F)cc2F)c1O c1(C(=O)NC(C(CO)NC(c2oc(CC)c(C)c2)=O)C)coc2c1COC2 c1(CC(C)N(C(CCN(CC)CC)=O)CCC(=O)NC2CC2)cccnc1 N1(C(C(=O)NC)=O)CCCN(C(=O)CC2CC(C(F)F)C2)C(C)C1 C1(CN(C(=O)CC2COCCO2)CC)CCCCN1C(=O)CCc1cscn1 C=C(C)c1cn(CC2COC(CNC(C34CC(C)C3C4)=O)C2)nn1 CC1CCC(C(=O)NCCC2CN(C(=O)C3=NNC(=O)C3)C2)C(=O)N1 N1(C(=O)OC(C)(C)C)CCC(CCF)(CNCC2CC2(F)F)C1 Cc1cc(C(F)(F)CC2CC2)cnc1Cl.n12cc(cn1)C1CN(C1)C(=O)C2 C(=O)(CC(C)C(=O)OC)NCc1c(C(=O)NCc2c(CC)n[nH]c2)cccn1 C1(C(=O)NC(CN(C(C(CC=C)C)=O)C)(C)C)Cc2cc(Br)cnc2C1 CN1CCCC2(CCN(c3cc(C(N4CCC(O)C4)=O)c4ccccc4n3)C2)C1 C1(c2ccc(C(=O)OC)cc2)CCCN(Cc2nnc(-c3ccccc3)o2)C1 N1(C(C2(SC)CN(C(=O)CCCc3ncco3)C2)=O)CCCC2(C=CCO2)C1 C1(CNC(c2c(CCC)nsc2N)=O)CC2CCC1N(C(C1CC1(F)F)=O)C2 c1(C(N2CC(CNC(C3N(C)C(=O)CC3)=O)C2)=O)nnc2ccccn12 C1(CC(=O)NC2CCC(F)(CNC(c3c(C)ncn3O)=O)C2)(OC)CCOCC1 N1(C(C2N(C(CC3(OCC)CCC3)=O)CC=C2)=O)CCCC(C)(C)CC1 C(=O)(N=c1ccn(CC)[nH]1)C1(CO)C(=C)C1.N1(C=O)C(CC2CCCO2)CC1C N1(C(C2=CC(C)CC2)=O)CCCC2CN(C(=O)CCn3cc([N+](=O)[O-])cn3)CC12 Cc1occc1C(=O)N(CCCOCCN(C(=O)C(c1ccccc1)O)C)C C12(C(N(C3CCCOC3)C)=O)CC1CN(C(c1cscc1Br)=O)C2 c1(OC)cc(O)c(CN2CCC(F)(C(=O)Nc3nc4c(s3)COCC4)C2)cc1Cl Cc1ccsc1CC(=O)NCC1CC(F)(CNC(=O)CCc2nncs2)C1 N(C(=NCCCCl)N1CCN(C(c2ccco2)=O)CC1)CC(CC)C(C)C C(CN=C(NCCCF)N1CCCC(OC(=O)N(C)C)C1)c1cccc(OC)c1 C1(C(CC(=O)O)NC(C2CCCN2C2CCCC2)=O)CCCC(=O)N1 CC1CCCN(C(=O)C(C2CC2)NC(=O)CS(C)(=O)=O)CC1 C1(NC(CC2CC(SC)C2)=O)C2CC(NC(c3ccc(Cl)cn3)=O)CC12 C(C1CCC(C)CC1)=C(C)C(N1CC(NC(c2c[nH]cc2C2CC2)=O)C(C)C1)=O C1(SC)(CNC(=O)NCCCNC(=O)Cn2cc(Br)cn2)CCCC1 C1(NC(C2C(C3CC3)C2(F)F)=O)CN(C(=O)C=CBr)C2(CCCCC2)C1 Cc1ccc(CCCNC(=O)CCn2cc(CNc3ccccn3)nn2)cc1 C#CCCCCCC(=O)NCC1CC2CC2N1C(c1ccc2cncn2c1)=O N12C3CCC1CC(C3)OCCS2(=O)=O.c1(C(=O)CC)cnc(OCC)nc1 c1(CNC(C2N(C(C(CC)n3cncn3)=O)CC2)=O)nnc(O)n1C CC1CC(NC(C2CCCCCC2)=O)CCN1C(c1cc(F)c[nH]1)=O Cn1cc([N+](=O)[O-])c(CSCC2C(Nc3ccccc3)CCCC2)n1 c1(SCNC(C(c2n(CC)nc(Br)n2)N(CC(C)C)C)=O)cc(F)ccc1F C1(C(C)C)CN(C(C2COCCO2)=O)CCN1C(=O)COc1cc(F)ccc1Br c1(C(NNC(=O)NC(c2sccc2C)CC)=O)cccc2ccccc12 S(=O)(=O)(CCC(F)(F)F)N1C2CC(C(=O)Nc3ccccc3Cl)C1CC2 c1(OC)cc(N2CC(NC(=O)Cn3nc(C)oc3=O)CC2C)c(Cl)cc1[N+](=O)[O-] C1(CCCNC(C23CCOCC2C3)=O)CCCCN1C(=O)CNc1nccs1 c1(C(=O)NCC2(F)CN(C(=O)NCCCl)C2)ccc(F)c2ccccc12 N12CC3CC(CC(C3)C1)NC2=O.c1(SC(C)C(=O)NC2CC2CF)ccccc1 c1(NCC(C2CCOC2)OC)nc2ccccc2nc1N1CC2CSCC(C2)C1 C1(CN(C)C(C2CC(C(=O)OCc3csc4nccn34)C2)=O)OCCCC1(C)C c1(NC(c2nc(NC(c3ccc(OC)o3)=O)sc2)=O)cnnc(O)c1Cl C1(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C)CCCCC1(F)F c1(C(=O)NC2CN(C(c3n(C)nc(C)c3Cl)=O)C(C)CC2)cc2ccccc2[nH]1 C1(C)(NC(C(CCC)=CCC)=O)CCN(C(=O)C(O)Cc2ccc(F)cc2)CC1 c1(C(=O)NCC(C2CC2)NC(C2COC2)=O)cc(Cl)c(Cl)s1 C1(c2ccn(C)n2)CCN(Cc2cc(C(=O)O)c[nH]2)CC1 Cc1occ(-c2ccccc2)c1C(N1CCC(N(C(=O)CC2CC23CC3)C)C1)=O CC(C)(CNC(N1CCC(CCO)C1)=O)Cn1cc(CCCC#N)nn1 Cc1cccc(NCC23CC2CCN3)c1C N1(C(c2ccc(SC)s2)=O)CCC2CN(C(=O)Cc3ccc(F)c(C)c3)CCC12 c1(C(=O)NC2CN(C(C(C)=C3CC3)=O)CC2C)ccc(Br)cc1[N+](=O)[O-] CC1CC(C(=O)NCc2ccc(C(=O)NC34CCCN(CC3)C4)s2)=NO1 C(C(=O)N=c1cc(-c2ccsc2)[nH][nH]1)(C(C)C)c1c(O)ccc(C)c1 CC(O)(CNC(=O)CCN1CCCC1)CNC(=O)CC1CC=CCC1 C(=O)(CCC(C)CN(C)C)NCCC(CCNC(c1nn(CC)c(C)c1)=O)C C(=O)(C(C#N)C(C)(C)C)N1C(C)CC(CNC(c2nc(OCC)sn2)=O)C1 N1(C(C=CC)=O)CCC(CNC(c2coc(Cl)n2)=O)C(C)C1 c1(C(=O)NC2C(COC)N(C(C3CC3OC)=O)CC2)oc2ccc(C)cc2c1C CC1CN(C(=O)CCSCC(=O)O)CC1(C)CNS(=O)(=O)CC1CCC1 N1(C(c2n(COC)ncc2)=O)CCN(C(C2CCCCC2C(N)=O)=O)CC12CC2 c1(CNC(CC(C)SC)=O)cccc(NC(c2ccns2)=O)c1 N1(C(c2nc(C)[nH]n2)=O)CCCCC1C(C)NC(c1coc(C2CC2)n1)=O CC1OCC2(CCC(NC(N3CC(c4cccc(Cl)c4)C3)=O)O2)C1C N1(C(CC2(COC)CC2)=O)CCC(NC(=O)CC23COC(C)(C2)C3)C(C)(C)C1 C1(C)(C(N(C)CC2(O)CN(C(C(c3cccc(F)c3)C)=O)C2)=O)CCSCC1 N1(C(C)C)CCC(NC(=O)C=CC2CCOC2)C1.C12CC(C1)C(=O)NC2 N1(C(C(COC)N(C)C)=O)CC2(CC(CNC(c3ccn(C)n3)=O)C2)C1 CCC(CC)C(=O)N(CCCNC(c1ccoc1)=O)CC.C12CCCC1NC2=O N1(C(C(C2CCCO2)OC)=O)CC(O)(C(=O)OCCN(C(C)(C)C)C(C)C)C1 c1(-c2cccc(NC(C)C(=O)C3CC3)c2)ccc2c(c1)COC(C)(C)O2 N1(C(c2ccc(F)cc2)=O)CCC2CCCN(C(c3cc4[nH]ccc4s3)=O)C2C1 C1(OC)CCCCC1C(=O)NC12CC(C1)N(C(c1ccc(C(N)=O)nc1)=O)C2 n1(CC)cccc1C(=O)NC(C1CCN(C(c2ccnn2C2CCCC2)=O)C1)C N1(C(Cc2c(C)occ2)=O)CCC(CNC(C2CC3CCC3C2)=O)CC1 C1(CNC(Cn2c(C)c(Cl)cn2)=O)C(C2CC2)CCN1C(=O)C(N=[N+]=[N-])C(C)C C(CCCCNC(=O)C(F)F)N(C)C(c1sccc1NS(C)(=O)=O)=O C1(OC)CC(CN(C(c2[nH]c(C)cc2C)=O)CO)N(C(=O)CC(=O)OC(C)(C)C)C1 C12(NC(CCOC)=O)COC(CNC(c3csc(-c4cccc(F)c4)n3)=O)(C1)C2 C1(CC(=O)NCC2(OC)CN(C(=O)C(F)=C(C)C)C2)CCCC(O)C1 N1(C(c2c(C)n(C)cn2)=O)CCC(NC(c2ccccc2F)=O)C(O)C1 C1(CNC(Cc2ncc(C)s2)=O)CN(C(c2cnn[nH]2)=O)C2(CCC2)C1 C1(C(=O)NC(c2cn(-c3ccn(C)n3)nn2)CCC)CC(O)(C2(O)CCC2)C1 c1(OC)cc(CN2CCC(NC(=O)Cn3ccnn3)C(F)C2)c(OC)cc1Br c1(C(N2CCC(NC(C3CCSCC3)=O)CC2)=O)ccc2cnnc(O)c2c1 Cc1nc2cc(C(N3CCC(CN(C)C(C4(n5ccnn5)CC4)=O)C3)=O)[nH]c2s1 CC1(C(N2CC(CNC(=O)C(=Cc3cccnc3)F)C2)=O)CC2(CCC2)C1 C(=O)(C(F)(CNC(=O)C=Cc1cn(C)nn1)C(C)C)N1CC(CCCCC)C1 Cc1cnc2cccc(C(N3CC(NC(=O)Cn4cncn4)CCC3C)=O)n12 c1(C(=O)NC(C2CCCN(C(CCC(=O)NC)=O)C2)C)ccc(F)c(F)c1F c1(N(C(C(CC#C)NC(c2cccc(CO)n2)=O)=O)C)cccc(C#C)c1 N1(C(C(COC)O)=O)CCN(C(c2c(C)ccn2C)=O)CC1CF N1(CC(C)NC(C(C=C)O)=O)CCN(C(C2(C3CC3)CCC2)=O)CC1 N1(C(C)=O)CCC(C)(NC(N2CCCN(c3cc(C(N)=O)ccn3)CC2)=O)CC1 c1(CC(=O)N(C)CC2COCCN2C(=O)C2=CSCS2)c(Cl)cccc1Cl N1(C(Cc2cc(COC)on2)=O)CC(NC(C2CC(C)=NO2)=O)C(C(F)(F)F)C1 n1(CCNC(c2cn(C(F)F)cn2)=O)ccc(C(=O)NCC2COC(=O)C2)c1 CC1=C(C)CC(C(=O)NCC(O)CC(=O)N(C)CC23CCC(CC2)CC3)CC1 C1(C(=O)NC2CC(NC(c3cn(CCC)nc3C)=O)C2)CCN(C)C(C)C1 c1(C(=O)NCC(CC=C)C(=O)NC2COC(C)(C)C2)c(C)nc2ncnn2c1C CN1CCN(C(=O)CCN(C(C2CC2c2ccccc2)=O)CC2CC2)C(CO)C1 C(=O)(CC(C)CC(F)(F)F)N1C(CN(C(C(CC=C)CC=C)=O)C)CCCC1 c1(C(c2n(C(C(=O)OC)C)nnn2)NC2CCCCC2)cc(F)c(OC)cc1Cl NC(CC(=O)N1CCCC(C(=O)O)CC1)C(F)F C(CC(C)(C)C)(C(=O)NCc1nc(C(C)C)no1)NC(CN(CCOC)C)=O N1(CC(=O)NC(C)CCCCNC(C2CC(C(F)F)C2)=O)CCCCS1(=O)=O C1(CNC(CCC)=O)CC(NC(=O)C=C(C)c2ccco2)CCO1 C1(CC(=O)NCC(O)CNC(c2cnoc2-c2ccco2)=O)CCCS1(=O)=O Cc1ncnc(C(=O)NC2CC=C(C(=O)NCC3C4CCCCCC34)C2)c1C Cc1ccc(O)cc1CCCC(=O)NC1CCC(n2cc(C3CCC3)nn2)CC1 Cc1csc(C=CC(=O)NCC(C(C)C)NC(=O)C=CCOc2ccccc2)n1 c1(C(=O)NCC2C(CNC(COC(CC)(C)C)=O)C2)cc(Br)n[nH]1 Cc1cc(C)c(C(N2CC(C)(CNC(=O)COCCC(C)C)C2)=O)c(Cl)n1 c1(C(=O)NCCCN(C(C(C)=C2CC2)=O)CC2CCCC2)c(Cl)cc(Cl)nc1N C(C(F)(F)CNC(=O)C(CC1CC1)NC(=O)COC(C)(C)C)OC c1(COC)cc(CC(=O)NCC2(C)CC(NC(=O)Cc3[nH]cnc3C)C2)no1 c1(C(=O)NC23CC(CNC(=O)Cc4ccco4)(C2)C3)cccc2nc[nH]c12 C1(NC(c2noc(CC)c2C)=O)CCCC12CN(C(=O)CC1COC(C)(C)C1)C2 CON(CCC(=O)N(C)C)C(=O)C(F)(F)CCn1cc(CC(O)C2CC2)nn1 C1(CCC)CN(C(C2(CCOC)CC2)=O)CCN1C(=O)CNC(N1CCCC1)=O C1(CCOC)CN(C(=O)CCC(=O)c2ccccn2)CCN1C(C1CC(F)C1)=O Cc1cc(F)cnc1C(=O)N(CCCCCCNC(=O)C(C)CC1CCCC1)C N1(C(CCOC2CN(C(C(C(C)C)O)=O)C2)=O)CCCC2CC1C2(C)C CC(C)CC(C(=O)NC(C)CNC(=O)Cc1coc(C(F)F)n1)N1CCCC1=O c1(CNC(=O)CN2CCC(C(F)(F)F)(CO)C2)ccc(N2CCCC2)cc1 c1(C(=O)NC2CCCCN(C(c3c(OCC)scc3)=O)C2)cnn2ccccc12 c1(C(N2CCN(C(COC(C)C)=O)C(C3CC3)C2)=O)cc2cn[nH]c2cn1 c1(NCC)cncc(C(=O)NCC2CC(F)CN2C(c2cc(C(C)C)[nH]n2)=O)c1 N1(C(CCSCC(C)C)=O)CCCC2(CCCN2C(C2OCCOC2C)=O)C1 c1(COCC)nnc(N2CCOC(CC(=O)NC)C2)n1CC1CCCO1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)C(F)(F)c2ccncc2)C1 C12CCC3CN(CC3C1)C(=O)CCSc1c(cccc1)CC(=O)N2.C1(CO)CC1 N1(C(c2cnc(C)s2)=O)CCC(C=CC(=O)NC2CC(=O)N(C)C2=O)CC1 c1(C(N(C)CC2CCCN(C(C(C)C#N)=O)C2)=O)cc2cccnc2cc1F C1(C(=O)NC(c2nccs2)CC)CCCN(C(C2CC3(CSC3)C2)=O)CC1 C1(CNC(c2cc(CC)nn2C)=O)CN(C(c2cnn3ccsc23)=O)CC1(C)C CC(CSc1ncccc1F)CC(=O)NCC1CCN1C(C1(CCF)CC1)=O C1(NC(C(CC)(C)O)=O)CCCCN(C(=O)COc2c(C)nc(C)nc2O)CC1 c1(N(C)CC2CCS(=O)(=O)C2)ncccc1S(=O)(=O)N(C1COCC1O)C c1(CC(=O)N(C(CCNC(C(C)(CO)OC)=O)C)C)c[nH]c2cc(Cl)ccc12 S(=O)(=O)(c1cc(C)ccc1C)NCC(=O)NC1CCCC(NC(C2(C=C)CC2)=O)C1 C1(C)(C(N2CCCC(N(C(C=CC(C)(C)C)=O)CCO)C2)=O)CCC(F)(F)C1 c1(N(CC(=O)N(C)CCNC(c2cc(Cl)nc(=N)[nH]2)=O)C)ccc(C#N)cc1F CCCCC(C)C(=O)NC1(COC)CCCN(C(c2c[nH]c(Br)c2)=O)C1 c1(NC(C)=O)cccc(C(=O)N(CCCN(C)C(c2cn[nH]c2)=O)C)c1 C(=O)(C(CC(N)=O)NC(C1CC1Cl)=O)N1C(C)(C2CC2)CC1 C1(C(=O)NCCNC(C=C(CC)C)=O)CCC(NC(=O)N(C)C)CC1 C1(CC(C(=O)NC(C)C)N(CC(CC)O)C2CC2)CC(C)(C)OC(C)(C)C1 N1(C(c2ccc(C#N)o2)=O)CCC(C2CC(NC(=O)Cc3ccc(O)nc3)C2)C1 N1(C(c2c(CC)n(C)nn2)=O)CCC(C)(C)C(C(=O)NCC2CC(F)C2)C1 CC1=C(C(=O)N2CCC(NC(C3(CO)CCCCC3)=O)C2C)C(=O)OC1(C)C c1(C(N2CCC(CC=C)C2)C(=O)NC(C)C)ccc2nc(C)ccc2c1 CCC(C(=O)NC(c1cn(C2COC2)nn1)C)C(F)(F)F C#Cc1ccc(OC)c(C(N2CCC(C)(CNC(c3cccs3)=O)C2)=O)c1 C1(NC(=O)C=CBr)COCCN(C(c2cccc(F)c2Cl)=O)C1 c1(C(=O)NC(CC)CN(C)C(c2cc(C)no2)=O)cncc(C(=O)OC)c1 c1(N(C2CCC(NC(=O)CCC34CCC(CC3)C4)CC2)C)nccc(C#N)n1 c1(CC)ccc(C(=O)NCCC(O)C(=O)NCc2nn(C)cc2CO)cc1 C(=O)(C(CC)C(F)(F)F)N1CCC(C=CC(N2CC(C#C)(N(C)C)C2)=O)CC1 C1(CC(=O)NC(c2nc(C(=O)NCC3CCCC(C)C3)co2)C)C(C)(C)C1(C)C c1(C(N(CC(C)(C)NC(C(CC)CN2CCCCC2)=O)C)=O)c(Cl)c(C)nn1C n1(CCC(N2C(CN(C(=O)COC3CCC3)CC)CCC2)=O)ccccc1=O Cc1cc(C(C)C(=O)NC2CN(C(=O)C(C)CCO)C2)cc(C)c1 c1(OC)cncc(CNC(=O)CN(C(=O)C(C)C#N)C(C)C)n1 C(C)(CC(=O)NCC1CCC(C(=O)NOCc2cccnc2)C1)OC C1(NC(C(CC)O)=O)CCOCC1NC(c1cccnc1N(C)C(C)C)=O c1(C(N2C(CCNC(c3ccnn3CCF)=O)CCC2)=O)cn2ccsc2n1 CC1(C)CCCCC(C(N2CC(NC(c3ncccc3O)=O)C2)=O)C1 c1(NC(C(Cc2ccccc2Br)NC(C)=O)=O)c(Br)nn(C)c1C N1(CC(=O)NC(C2CCCCC2)C#C)CCN(C(C2OCCOC2C)=O)CC1 c1(C(=O)NCC2(NC(CCCCC=C)=O)CC2)ccc2c(Br)cnn2c1 C(=O)(C(C(C)C)n1cncn1)NCCC(=O)C(C)(C)C.CCCN1CCCC1.OC C1(OC)CCCC1C(N1CCCC1C(C)(C)NC(=O)C=CC=C(Cl)Cl)=O N1(C(COCCC)=O)CCC2CC2(NC(=O)Cc2cc(OC)ccc2CC)CC1 c1(C(=O)NC(CCOC)CNC(=O)CCCc2nccs2)cccnc1Cl c1(C(=O)NC2C(NC(c3n(C)c(S)nn3)=O)C2)cnc(O)c2cccnc12 C1(CC)(Cc2cccnc2)CCN(C(=O)Nc2n[nH]c3c2COC3)CC1 CC1(CNC(=O)Cc2cscn2)CCCN(C(=O)CCC2NC(=O)NC2=O)C1 c1(NC(C(C)OC)=O)cccc(S(=O)(=O)N2CCSC(c3ccccc3)C2)c1 c1(C(N2C(C(C)C)CN(C(C3CC3C(N)=O)=O)CC2)=O)cc(=O)n2ccsc2n1 Cc1c(C(N2CCCCCC(NC(=O)C(C)(C)F)C2)=O)sc2ccc(Cl)cc12 C1(NC(Cn2ncc(C)c2)=O)C(C)CCN(C(c2cc(O)cc(N)c2Cl)=O)C1C c1(-n2cc(C3N(C(Cc4occ(C)n4)=O)CCC3)nn2)ccc(C)c(C(=O)O)c1 Cc1ccc(C(=O)NC(C(=O)N(C2CCOC2)CCO)C2CC2)o1 C=CCC(CC)N=c1nc(N(C)Cc2noc(C)n2)c2cnn(C)c2[nH]1 c1(C(c2n(CCC)nnn2)N(CC)Cc2ccon2)ccccc1Br c1(C(=O)NCC2C=CC(NC(CCCCOC)=O)C2)cc2sc(C)cc2s1 c1(CC(=O)NC(CCN(C(C2C(=C)C2)=O)C)C)sc(C2CC2)nc1C Cc1cc(=NC(=O)C2CCCC23CCN(C(=O)CCS(C)(=O)=O)C3)[nH][nH]1 N1(C(C=COCC)=O)CC(CNC(c2ccnn2CCF)=O)CC1(C)C C1(C(=O)NC(CC)C)CC2(CCN1C(C1C=CC1C(=O)OC)=O)CC2 N1(C(CC2C(C)OC(C)C2)=O)CCCC(N(C)C(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(NC(C(c2ccc(C)cc2)C)=O)CN(C(=O)CC2CN(C)C2)CC(C)(C)C1 C12(CNC(C3CCCC3)=O)CC(CCO1)N(C(c1cccc(CO)c1)=O)C2 c1(NC(C(C)O)=O)cccc2c1C1CN(C(=O)COc3ccccc3Br)CC1O2 C1(NC(CCc2ccn(C)n2)=O)CC2CC(NC(c3cncs3)=O)C2C1 C1(C(N2CCC(CNS(C)(=O)=O)C2)C(=O)NCc2ccco2)CCOC1(C)C N1(C(c2cc(CC)cc(N)c2)=O)CCC(C2CC(NC(=O)C(C)(Cl)Cl)C2)C1 c1(NC(NC(C(C2C(C)(C)C2)C2CC2)=O)=S)cnn(CCF)c1 CN1C(=O)CCCC1C(=O)NC1CC2CC(NC(c3cnns3)=O)C1C2 CCCC(C(=O)NC1CCN(C(C)C)C1=O)NC(=O)Cc1cnn(C)c1 C1(C(=O)NCC(C2(C)OCCO2)C)(CC)CCN(C(=O)C=C=C(C)C)C1 C1(N(C(c2cnsc2)=O)CC)CCCN(C(C2CC23CCSCC3)=O)CC1 c1(C(=O)NC2CC3CC(NC(=O)CCc4cscn4)C2C3)ccc2nncn2c1 C(C(C)(CC)C(=O)NC(c1cccnc1)C)NC(CCC(=O)NCC)=O N1(C(C2(SC)CC2)=O)CCC(F)(F)C(CNC(=O)CCCC2CCC2)C1 C(CCC(=O)NC(C(=O)NCCCSC)C1CCSC1)OCCOC c1(C(=O)NCC2(F)CCCN(C(c3nc(=N)[nH]cc3)=O)C2)ccnc2cc[nH]c12 N1(C(c2nc(COC)oc2)=O)CC(C)CN(C(c2cc(Cl)no2)=O)CC1C C1(C(=O)NCc2c(C(=O)NC(CO)CO)occ2)CC(F)(F)CS1 c1(C(C(=O)NC2CC(C)(NC(C(CC)F)=O)C2)(F)F)ccccc1C C(=O)(C1CCCn2ncnc21)NCC1CN(C(C(C)C)=O)C1 C1(C(N2CCC(CNC(c3cccc(OC(F)F)c3)=O)C2)=O)CC2CC1CO2 N1(C(c2cccc(Cl)c2OC)C(=O)NCCCCCC)CC2OC(=O)N(C)C2C1 N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(=O)CC2CC=CCC2)CC(C)C1 N1(C(C2(CC=C)CCOCC2)=O)C2CCC1CN(C(=O)CCCCCCC)C2 C12(CNC(CNC(CC)=O)=O)CCC(CN1C(=O)Cc1csc(C(C)C)n1)C2 C(=O)(C(C)(C)C(=O)NCC1C2CN(C(=O)CC3COCCO3)CC12)OCC CCCC(C)(CC)C(=O)N1CC=C(C(=O)NCC(O)(COC)CO)C1 C1(CCC)CCCN(C(C23CC2CN(C(=O)CC(C)SC)C3)=O)CC1 c1(C(=O)NC(C2CCCC2)CNC(C2C=CCC2)=O)ccc(C(F)(F)F)cc1 c1(C(=O)NC2CCCN(C(c3c(C#C)c[nH]n3)=O)C2)cnc(C)cc1Cl Cc1ccc(CC(=O)NC2CCC2CNC(C2CCCSC2)=O)cc1 C1(F)(CNC(C2CCCO2)=O)COCCN(C(=O)C=CCN2CCOCC2)C1 C1(C(=O)NC)CC(N)C1(C)C.c1(C(=O)C2CC2)ccc(OCCCNC=O)cc1 c1(C(=O)NCC(CN(C(C(CC)N(C)C)=O)C)O)ccc(OC)c(C)c1 Cc1ccc(CNC(CCN(C)C)C(C)C)c(I)c1 C(CC(O)C(=O)NC1(Cc2ccccc2NCC(=O)NCC2CC2)CC1)N(C)C c1(C(C(=O)N(CCNC(=O)CN(C)C(N)=O)CC)C)c(F)cccc1F N1(C(Cc2c(N)cc(F)cn2)=O)CC(NC(C2CC(=C3CC3)C2)=O)CC(F)(F)C1 O=C(CCCCNC(C1CC(CCO)C1)=O)NCc1nocc1C(=O)O CC(CC(C)(c1nnnn1C1CC(F)(F)C1)N)C(F)F.C(C(C)(C)SCCO)S CC1CCN(C(=O)Cc2ccnc(O)c2)CCN1C(=O)COc1ccsc1 Cc1nn(C)cc1C(=O)NC(CCN(C)C(C1CCC(C)CC1)=O)C(C)C c1(C(=O)NCC2C(NC(c3noc(CC)c3C)=O)CC2)cc(C)cc2ccoc12 Cc1cccc(CN(C(=O)CCN(CCCO)C(c2cccnn2)=O)C2CC2)c1O Cc1cc(C(N2CC3(CC(CC(=O)NC(C)C(C)N(C)C)C3)C2)=O)ccc1O N1(C(CCc2ccc(C)cc2)=O)CCC(C(=O)NCC2CCC2CO)=C(F)C1 Cc1ccc(C(=O)NCC2CCCCC2NC(C23CC(F)(C2)C3)=O)c(C2CC2)n1 C1(C2CN(C(=O)C=CC=C(Cl)Cl)C2)(NC(C2CC(C(F)F)(OC)C2)=O)CC1 N(C1CCCc2ccoc21)C(C1C2CN(C(C3C4CN(C)CC43)=O)CC21)=O c1(N2CCC(N(C)CC)CC2)nc2c(c(=NCC3CC(O)CCO3)[nH]1)CCC2 C=CCC(C)(O)C(=O)NC(c1ccccc1)C(=O)NCCC(O)C(F)F c1(C(=O)NCC(CNC(CC2N(CC)CCOC2)=O)(C)O)cc(F)ccc1F C1(C(N(CC(C)N(C)C(c2coc(O)n2)=O)C)=O)COCOC1 CCC(C(=O)N1CC(N2CCN(C(=O)Cn3nnc(C)n3)CC2)C1)C(C)(C)CC C(C(C)(C)CNC(c1cn(C2CC2)nn1)=O)N1C(=O)CCC1.C(C)(=O)OCC c1(NCC(N2CC(CCCCNC(C(CSC)OC)=O)C2)=O)ccc(Cl)c(Cl)c1 CCC(CC)C(C(=O)NC(CC)CC(N1CCC(O)C(CO)C1)=O)OC C12(C(=O)NCC3N(CC)CCC3)CC(C(=O)NC3CCNC3=O)(C1)C2 Cc1c(C(N2CCC(CN(C)C(c3ccc(Cl)cc3)=O)CC2)=O)cccc1F Cc1cc(F)cnc1C(=O)N(C1CCN(C(C2CC(C)(F)C2)=O)CC1)C C1(C(=O)NCCC2CCCCN2C(=O)C=Cc2cscn2)CCOCC12CCC2 Cc1ccc(C(C)C(=O)NC2CC(CNC(C34CC(C)(C3)C4)=O)C2)s1 c1(C(=O)NCCN(CCC)C(=O)SC2(CC)CCC2)oc2ccccc2c1CC Cc1nc(NC2CCN(C(=O)C(C3CCOCC3)F)C(C)C2)cc(C(F)(F)F)n1 N1(C(C2N(C(c3c(NC)cccc3)=O)CCCC2)=O)CCN2CCCCC2C1 c1(C(=O)NC(C2CCN(C(=O)C=CC3CCCC3)C2)C)ccc(Br)cc1O c1(OC)cc(C)c(C(=O)NC(CNC(=O)C2=NNC(=O)C2)CC(C)C)cc1OC C1(O)(CNC(C(C)n2ccnn2)=O)CCN(C(=O)C=CC2CCCC2)CC1 c1(OC)ccc(CCCNC(N2CCCC(CC(=O)OC(C)(C)C)C2)=O)nc1O c1(C(N2CCC(C)C2C(N2CCS(=O)CC2)=O)=O)cc(O)cc(F)c1 C1(CNC(CCc2n(C)cnc2)=O)CCC(C)(C)CN1c1cc(=O)n(C)cn1 c1(C(N2CC3=C(CN(C(CCN(C(C)=O)C)=O)C3)C2)=O)ccc(F)c(C)c1C#N S(=O)(=O)(c1ccc(N2CCOC(C(N)=O)C2)cc1Br)NCCC1CC(C)(C)OC1 CCC(CCC(=O)NC(C)(COC)CC)NC(C1CC1c1ccco1)=O c1(C(=O)NCC2CCCN(C(C(CC=C)C(C)C)=O)C2)cc(C)c2[nH]cnc2c1 C12(C(=O)NC3(CC=C)CN(C(=O)OC(C)(C)C)C3)CC(C)(C1)OC2C N1(C(c2c(C)ccs2)=O)CC(C(N2CCSCC2CO)=O)C2(CCC2)C1 O=C(CCN1C(=O)CCc2cc(F)ccc21)NC1CCN(C(=O)CO)C12CC2 c1(C(=O)NCC(O)CNC(C2CC(F)(F)C2)=O)cc(Cl)ccn1 Cc1cc(C(N2CC(NC(c3ccc(C)s3)=O)CC(C)C2)=O)n2ncnc2n1 N1(CCNC(C2CCC2OC)=O)CCOC(CNC(C2(C(=O)OC)CCCO2)=O)C1 C1(CC)C(C(=O)N(C)CCC2CCCCC2)CCN1C(C1COCC1C(N)=O)=O C1(C(=O)Nc2ccc(CC)cc2)CCC(C)N(C(=O)Cc2cc(F)ccc2F)C1 C(=O)(C1=CCCCO1)N1CCC(NC(c2c(C)nn[nH]2)=O)(CF)C1 c1(N)ccnc(N2CC3CC3(CO)C2)n1.CN(C)CCOC(F)F Cc1cc(C(=O)N(C)CC2CCCN2C(c2cscn2)=O)ns1 CCCCC(C(=O)N(C)CCOCCNC(=O)Cc1cncn1C)C(C)C N1(C(=O)COCCCF)CCN(C(C2CC3(C2)CC3F)=O)C(c2ccccc2)C1 c1(C(=O)NCCN(CC(C)O)C(c2cc(C(C)C)nn2C)=O)cnn2c1OCC2 C1(CC(C)NC(=O)CC2(O)CCC2)CN(C(=O)COC2CCC2)C1 CC(C)C(C)(O)C(=O)N1CC(C(=O)NCCNC(=O)C(N2CCOC2=O)C)C1 N1(C(CCC(C)OCC)=O)C2CCC1CC(N(C(=O)C(=CC1CCCC1)C)C)C2 N(C(=NCc1ccccc1)NCC(c1cn(C)cn1)(C)C)CCOCC=C Cc1nccn1CCNC(C1(NC(=O)C(=O)NC(C)C)CC1(C)C)=O Cn1c(C(=O)NC2CC2CNC(C2CC=CCC2)=O)nnc1S c1(NC(C2CCCN(CCCCCC(=O)OC(C)C)C2)=O)c(F)cc(Cl)cc1Br c1(N2CC(CNC(CC(C)n3cccn3)=O)OCC2)ncnc2[nH]ccc12 C(=O)(CCC(CF)CF)N1CC2CC(CNC(C(C)(C)N3CCCCC3)=O)C2C1 C#CCCCCCCC(=O)NC1CCCN(C(=O)CC(O)CCC)CC1 C(C(O)CC(=O)NC1CCC(=O)NC1)NC(C=C(CC)CC)=O C#CCC(C(=O)N(CCC)CCNC(c1sc(SC)cc1C)=O)C1CC1 C(N=c1[nH]c(=N)[nH]c(=NCC(F)(F)CC2CC2)[nH]1)C1N(C)CCOC1 c1(C(=O)NC(C2CCCCC2)CNC(C2C(C)C2)=O)nc2cncnc2nc1O CC(C)C(C)C(=O)NC1CCOC1C1CCN(C(C2(O)CC(F)(F)C2)=O)CC1 c1(C2N(C(CCNCC(C)C)=O)CCOC2)ccc(F)c(Br)c1 C12(CNC(C3CC34CCOCC4)=O)CCCC1CN(C(c1sccc1Cl)=O)C2 S(=O)(=O)(c1ccc(F)cc1)NCCCC(=O)NC1CN2CCNC1C2 N1(C(C(C)C2CCCO2)=O)CCOCC(NC(=O)COC2CCOCC2)C1 C1(c2nnnn2C2CC2)(NC2CCCC(C(=O)OC)C2)COCC(C)(C)C1 Cc1cc(=NC(=O)C(=O)N(C2CCSCC2)C)[nH]n1C(C)CN(C)C N1(C(c2cc(CCC)on2)=O)CC(NC(=O)CC(C)N(C)C)CCC1C CCC(C)C(C(=O)NCC1CCC(C(N2CC3CCC(C3)C2)=O)C1)N(C)C c1(C(=O)NC(C(C)NC(C2C(CC(C)C)C2)=O)CO)ccc(N2CCCC2)c(F)c1 c1(C(=O)NC2CC(NC(C3CN(C(=O)NC)C3)=O)C2)cc2c(=O)cc[nH]c2s1 C1(C(=O)NCCN(C(c2ccc(CC(C)C)nc2)=O)CC)CCS(=O)(=O)N1.C1(C)CC1 N1(C(C(F)OC)=O)CCN(C(=O)CCN(C)C)C(C(C)C)C1 C(=O)(C1=C(F)CN(C(=O)COCC(C)(C)C)CC1)NCCC1CC(C)C1 Cc1ccc(NC(C2OCCC2CNC(=O)C(C2CCCCC2)=O)=O)cc1F Cc1ccc(C(=O)NCC2CCCC(NC(c3ncoc3C3CC3)=O)C2)nc1O N1(C(CCC(=O)NC)=O)CC(CO)C2(C1)CN(C(=O)Cc1ccccc1)C2 c1(C(N2CCC(O)(CNC(C(C(C)C)SC)=O)C2)=O)cccc2cc[nH]c12 N#Cc1c(NC2CC(F)CN(C(=O)C3=NNC(=O)CC3)C2)cccc1Cl C1(C(=O)NC(c2nc(C)no2)CC)CN(C(=O)C(CC)SC)CC1CC C(C(F)C(=O)N(C1CN(C(=O)Cc2nnc(C)o2)C1)C)OCC CCCCC(CC)C(=O)N1CC(CN(C)C(c2ccc(F)o2)=O)C1 C(CC(=O)N1CCCC(c2nnc(C3CCC3)n2C(C)C)C1)(C(=O)O)NCC c1(OCC(=O)NC2CCN(C(c3cc(CC)no3)=O)C2)ccc(Cl)cc1Cl N1(C(C2CC(C)OC2)=O)CC2(CCN(Cc3cnon3)CC2)C1 C1(C(=O)NCCC2CCN(C(C3(C)CCCCO3)=O)CC2)CCC2(CCC2)CO1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCCC2C)ccc([N+](=O)[O-])cc1Cl C(=O)(C1=CS(=O)CCC1)NCC1(F)CCCN(C(CC(C)C)=O)C1 Cc1ccc(NC(=O)CC2C=CC(NC(C3CCCC34CCC4)=O)C2)c(O)n1 c1(OC)cc(C(=O)NC(c2ccc(NC(C)=O)cc2)C)ncc1Br c1(NC(c2sccc2NCc2ccc(Br)o2)=O)cc(F)c(F)c(F)c1F C1(N(C(C2(CSC)CC2)=O)C)CCN(C(=O)CN2CCC(OC)C2)C1 N1(C(C=CC)=O)CCN(C(c2conc2Cc2ccccc2)=O)CCC1C N1(C(C2CN(C(CC=CC)=O)CC23CC3)=O)CCC(O)C(C)(O)C1 C12(CCNC(c3c(C)nc(COCC)s3)=O)CCC(C1)N(C(C1CCOC1)=O)C2 C1(C(=O)NCC2(C(C)(C)O)CN(C(C(C(CC)C)=O)=O)C2)CCn2cncc2C1 CCCCC(C)CCC(=O)N1CCCCC1C(=O)Nc1cccc2c1OCO2 CC1CN(C)CCC1N(C)C(C1CCC(CNC(=O)CC(F)(F)F)O1)=O c1(OC)ccc(C(F)F)cc1C(=O)NCC12CC1CN(C(C1CC=CCC1)=O)C2 C1(NC(C2(SC)CCC2)=O)COCCN(C(c2ccnc(OC)n2)=O)C1 N1(C(C(C(CC)CC)C)=O)CCC(NC(c2cnc(O)c(Cl)c2)=O)CC(C)(C)C1 CC(C)(C(=O)NC1CCCC(CNC(C2CC3(CCO2)CC3)=O)C1)S(C)(=O)=O C#Cc1cccc(C(=O)NC2CCCCC2(C)CNC(C23CC(F)(C2)C3)=O)c1F C=C=C(C)CC(=O)N1CCC(CCNC(=O)CN2CC3CC3C2)CC1 NC1CC2(CNCCS(=O)(=O)CSC)COC1C2 C1(CCC)CN(C(c2ncoc2C)=O)CCN1C(c1cc(C(F)F)nn1C)=O C(=O)(CN=c1ncnc2[nH][nH]c(Br)c1-2)N1CC(CSC)C(C(F)(F)F)CC1 C1(C(=O)NC(C(C)NC(c2[nH]nnc2C(F)F)=O)C)CC2(CCO1)CC2 c1(OC)ccc(C(N2CC(C)(NC(C3CCCC(F)C3)=O)C2)=O)cc1 Cc1cc(=NCCc2ccc(C#N)cc2)[nH]cc1S(=O)(=O)NC1CC12CCOC2 Cc1ccc(C(N2CC(NC(=O)CCCc3ccc(Br)cc3)C(F)C2)=O)c(C)c1 CC1(C)CCC(CO)N(C(C2CN(C(=O)Cn3cnc(=N)[nH]3)CC2(C)C)=O)C1 C1(C(=O)NCC(CNC(=O)C(c2cccnc2)O)CO)CC12CCSCC2 CC1(C)OC2(CNC(C3CC3F)=O)CC1(NC(=O)C1CC1)C2 N1(C(CSCCCC)=O)CCN(C)C(CNC(=O)COC2CCOCC2)C1 N1(CCc2cc(CC)on2)C(C)CC(C(F)(F)F)C1C C1(C(=O)NCC2C(NC(CNC(=O)OCC)=O)C2)CC2(CC(=O)N2)C1 C1(NC(C2(COC)CC(F)(F)C2)=O)CCN(C(c2sccc2F)=O)CC1O C(=O)(C(O)CCCc1ccccc1)N(CC(C)(C)NC(C1N(CC)CC1)=O)C N1(C(C(CC=C)C)=O)CC2OCCN(C(c3scnc3-c3ccccc3)=O)C2C1 C=CC(CC(=O)N1CCC(N(C(=O)CN2CSCCSC2)C)C1)c1ccccc1 c12cccn(c1=O)CC(=O)NCC(C)NC2=O.c1(OC)cccc(C(=O)OC)n1 C1(CNC(COCCCCC)=O)C(CC)CCN1C(c1cocc1C)=O C#CCCCC(C)C(=O)N1CCCC1C(=O)NCCc1ncc(C)o1 c1(OC)ncc(Cl)cc1C(=O)NC1CC(CNC(=O)C(C)c2ccco2)CC1O c1(C2(C(N3C4C(NC(CCSC)=O)C(C4)C3)=O)CC2)ccc([N+](=O)[O-])c(C)c1 O=C(CC1=CCOCC1)N1CC(O)CC1C(N1CCCC(CO)CC1)=O C1(NC(c2cc(SC)oc2C)=O)CCSC12CN(C(=O)Cc1sccc1C)C2 N1(C(CC(C)C)=O)CCN(C(=O)C(CC(C)C)Oc2ccccc2)C(CO)C1 C1(N(C(=O)Cn2cc(C(F)(F)F)cn2)CCC)CCCCC1C N1(C(C=CC)=O)CCCC(C2CCN(C(=O)C(CC3CC3)CC3CC3)C2)C1 C1(C(=O)NCCOCCC2CCC2)CCN(C(c2ccc(C3CC3)o2)=O)C1 C(C(C(C)(C)C)NC(=O)CCc1ncccc1C)NC(C(=O)NCC)=O CCC(C(=O)N1CC2CCC2(CNC(c2nscc2C)=O)C1)C(C)C CC1OC2(C)CC1(C(N1CCC(CNC(c3ccnc(F)c3Cl)=O)C1(C)C)=O)C2 C1(N(C2(CC)CCC2)C(C2CCC2)=O)CC2(CCN(C(=O)CC(C)C(F)(F)F)C2)C1 c1(C(N(CCC(C(C)C)NC(COC(CC)C)=O)C)=O)ccnc(F)c1OC c1(OC)ccc(C(N2CCC(C)C2C(=O)Nc2cccnc2C)=O)cc1O c1(NC2C3CN(c4nc(C)c(Br)cn4)CC2CC3)ccc(S(C)(=O)=O)cc1 c1(CC)nc(O)c(C(=O)NCC2CN(C(=O)CC3CCNC3=O)C2)cc1C N1(C(C(C)N(C)C)=O)CCC(NC(=O)Cc2cncc(Br)c2)C(F)C1 C1(CNC(C(C)SC)=O)CCN(C(=O)CCNC(=O)CO)CCC1(F)F C(C(O)CC(=O)N1CC(F)CC1CNC(c1cc(C(F)F)no1)=O)N(C)C C1(C(N(C)Cc2noc(C3CC3)n2)=O)CC2(CCO1)CC2.C12CN(CCO1)C2=O N1(CCCCOC(C)C)CCCC1CNC(C1CCCN1CC(C)C)=O C1(C(=O)NCCC(C)(C)OC)CCCC(NC(=O)C=Cc2cccc(C)c2)CC1 c1(CC)cc(C(N2CC(NC(c3cc(F)c[nH]3)=O)C(F)C2)=O)cc(C)c1 c1(C(=O)NC2CCN(C(C3(C)CCOCC3)=O)C2)ccnc2ccc(N)cc12 O=C(C(F)C(F)(F)F)N1CC(c2ccc(COC3CCCOC3)cc2)C1 N1(C(C(C)C)=O)CC(NC(C2OCC2(C)C)=O)CC(C)(C)C1 c1(CCCC(=O)NCC2CC(F)(CNC(CC(=C)Br)=O)C2)nnc(C)n1C c1(OC)c(Cl)ccc(C(N2CCCN(C(=O)CC3C=CCC3)C(C)C2)=O)c1F C1(NC(C(C)NC(C)=O)=O)CC2C(CNC(=O)C(c3cccc(O)c3)C)C2C1 c1(C(=O)NCC2(CCNC(C(CC)SC)=O)CC2)nnn2c1CCC2 c1(CC)cccc(C)c1C(=O)Nc1ccc(Cl)nc1NS(=O)(=O)C(C)C C(=O)(CCCCCC(C)O)NC1CCC(CNC(c2cc(CC)nn2C)=O)CC1 C1(C(=O)NCC=CCC(=O)NCC(CO)OC)CNC(=O)N1 C1(CNC(C2C(C=C)C2)=O)CC2(C1)CN(C(=O)CC1(CO)CC1)C2 c1(C(=O)NCCC(C)N(c2cnccn2)C)c[nH]nc1-c1cnn(C)c1.C1CS1 c1(C(=O)NCCCNC(CC2CC(C(C)C)OCC2)=O)cc(F)c2[nH]nnc2c1 c1(C(=O)NC2C(NC(c3c(CC)nns3)=O)CC2)ccccc1N(C)C N1(C(CCS(N)(=O)=O)=O)CCC2(CC1)COC(CNC(=O)COC1CCC1)C2 CCC1=C(C(=O)NCC2(O)CC(NC(=O)C(C)(C)CC#N)C2)CCCO1 C1(C)(C(N2CC(CCC)C(NC(=O)C(C)(O)C(F)(F)F)C2)=O)CCC(=O)N(C)C1 C(=O)(C(CN(C)C)C(C)C)NCC1C(CC(N2C(CC)(CC)CC2)=O)C1 c1(C(N2CC(O)CC2CC(C)C)C(=O)NCCOC)c(Cl)ncn1C c1(C(=O)NC2CC3CN(C(COCCC)=O)CC32)cccc2c1CNC2=O N1(C(c2c(CC)nco2)=O)CCOC(C(C)NC(c2ccccc2C2CC2)=O)C1 CC#CCCC(=O)NC1CCC(C(=O)NC(CNC(=O)C(C)C)(CC)CC)CC1 c1(C(N(CCC(C)NC(c2n(CC(C)C)ncc2)=O)C)=O)ncnc2c1CCC2 C1(C)(C(=O)NCCC(NOC)=O)CCN(C(=O)C=C(C)c2ccccc2)CC1 CC1OC2(C(N3CC4CC(NC(c5cnnc(O)c5)=O)C3C4)=O)CCC1CC2 C(c1nc2ccccc2o1)=CC(=O)NC1CCN(C(C=C(CC)C)=O)CC1CO c1(SC(CC)CN(C)C)nnc(-c2ccc(OC)cc2)n1CCC#N N1(C(c2c(SC)scc2)=O)C2CCC1C(CNC(=O)C(C)CC(F)F)C2 Cc1ccc(CNC(=O)CCN(CCCO)C(c2cccc(F)c2C)=O)cc1F n1(C(C)C)ncc(F)c1C(N1CCOC(CN(C)C(C2CC2F)=O)C1)=O c1(C(N2C(CNC(C3CCCO3)=O)CC(C)(C)C2)=O)cc(Br)c2c(c1)OCO2 C12(C(N3CC(CC)N(C(=O)C(F)(F)CC(C)C)CC3)=O)CCOC1CCOC2 N1(C(C(C(C)C)OCC)=O)CC2CCC(C1)N2C(=O)COc1ccc(C)cc1F N1(C(c2cnc(CC(C)(C)C)s2)=O)CCC(C)(NC(c2n[nH]cc2C2CC2)=O)C1 N1(C(CCC(C)OC)=O)CCN(C(c2ccc(C)cc2N)=O)CC1C1CC1 c1(CNC(C(CCC)C)=O)c(C)nn2c1CN(C(C1(c3cccs3)CC1)=O)CC2 c1(C(=O)NCCC2CCC(NC(Cc3cc(C)on3)=O)C2)c(Cl)ccc(F)c1C N1(C(C2N(CC)CC2)(C)C)CCC(C)(CC(=O)NCC(n2ccnn2)C)C1 N1(C(c2c(C)nccn2)=O)CCCC12CCCN(C(=O)Cc1ccc(Cl)cc1)C2 C1(COCC)(NC(=O)Cc2occc2C)CCN(C(=O)C=CSC)CC1 CCC(C(=O)NCC1(NC(C2(C)CCCCC2)=O)CCOC1)C(C)(F)F C1(CC(=O)N(C(CC#C)C)C)CC(C)N(C(=O)CSCCC)C1 C1(C(=O)NCC2C(NC(CCC(=O)OC)=O)C=CCC2)CC(F)C(=O)N1C C1(C(=O)NC23CC(C)(C2)C3)CCCN(C(=O)CC2CCCN(C(C)C)C2)C1 C12(NC(C3N(C(=O)OC(C)C)CCC3)=O)CC1CN(C(=O)CC(O)CN(C)C)C2 C1(F)(CNC(C2CCCN(C(C)=O)C2)=O)CCCN(C(=O)CCC(C)C#N)C1 CC(C)CN=C(NCC(Cc1ccccc1Br)CO)NC1CCCC1(F)F C=Cn1nccc1C(=O)NCC1CC(NC(=O)CCNC(=O)CO)C1 C1(O)(C(=O)NC(CCC)CNC(c2c[nH]nc2C(F)F)=O)CCC(C)(C)CC1 C1(NC(C2CC(O)(CC#C)C2)=O)CN(C(=O)Cc2ccsn2)CC(C)(C)C1 C1(CNC(=O)CCc2cncs2)CC(CNC(=O)CN2CCSCC2)CO1 C1(NC(CCc2cc(C)on2)=O)CCN(C(=O)CC2CCC=CCC2)CCC1CO c1(C(C(=O)NC2(CCNC(C3CCCC(F)(F)C3)=O)CC2)O)cc(Cl)cc(Cl)c1 c1(C(=O)NCC2CC(NC(=O)CCF)C(O)C2)cccc2c1COC2 C1(C(C)(O)CNC(=O)CCc2cnco2)CCCN(C(=O)CP(C)(C)=O)C1 c1(C(N2C(CCNC(c3n(C)ncc3)=O)COCC2)=O)cnc2c[nH]nc2c1 CC1CCC(NC(=O)CCC2CC(C)(C)CO2)CN1C(=O)CCn1cncn1 Nc1cc2ccccc2cc1C(=O)NCC(O)CNC(=O)C=CC1CCC1 C1(NC(CSc2cn(C)nc2)=O)CC2(C1)CC2C(=O)NC12CC(F)(C1)C2 N12CCCC3C1CCCN3C(=O)C=CC2=O.c1(C(=O)NC)cc(OC)ccc1F CC(C)CC(CNC(C1(O)CC(C)(C)C1)=O)NC(=O)CCC(C)N(C)C c1(OC)ccc(O)cc1C(=O)NC1SCCC1C C1(C2CC2)(CNC(C(CCCC)N(C)C)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)C1 OC1CC2(CC(NC(c3sccc3Br)c3nnnn3C3COC3)C2)C1 N1(C(c2ccc(C)c(C)c2N)=O)CC23CCCCC2(C1)CN(C(C1C=C1C)=O)C3 c1(C(C)C)ccc(CN2CC(F)CC2C(=O)Nc2cc(C(F)F)cs2)cc1 c1(OC)cc(C#N)ccc1CNc1c[nH]nc1C(=O)NC(C1CCOCC1)C CC(CCCNC(c1cc(Cl)no1)=O)NC(=O)CCc1nc(C(F)(F)F)n[nH]1 C1(NC(CC(CCC)CC)=O)CC2CCCC(C1)N2C(C1CCCCC1C)=O C(c1ccccc1C)=CC(=O)NCCNC(c1c(C)cn(C)c1)=O C1(NC(CCOCC)=O)CCC(C)(NC(=O)C(F)Cc2ccccc2)CC1 N1(c2cc(NCCC(c3ccc(F)cc3)C)ncn2)CCc2ncn(C)c2C1 CCCC(C)(CC)C(=O)N1CC2CC1(C(=O)NCC(CC1CC1)OC)C2 C=C1Cn2c(C(N3CCCN(C(c4c(C)ncn4O)=O)CC3CO)=O)nnc2S1 c1(CC(C(=O)NC(CNC(CCCOC(C)C)=O)C)O)ccc2ncccc2c1 C1(CNC(=O)CCCCCCn2cc(CO)nn2)CCCC2(CCOCC2)O1 c1(C(=O)NCC#CCNC(C(COC)N(C)C)=O)ccc2c(c1)COC2 C12(C(=O)NC(C)CCC3CCCO3)CC(CO)(CN1C(c1ccns1)=O)C2 C1(NC(C(C)=C(C)C)=O)CC2(CCN(C(c3cccc(C4(C)CCO4)c3)=O)C2)C1 C1(C(=O)NC(c2c(C)n[nH]c2C)C)CN(C(c2cocn2)=O)CC(C)O1 C1(C(N(C(C)C)CCNC(c2ccsc2)=O)=O)C2CN(C)CC12 C12(CNC(C(c3ccc(OC)nc3)(F)F)=O)CC(C1)C(NC(C1CCC1)=O)CO2 c1(CC(=O)NCC=CC(=O)NCC(C)(C)O)cccnc1O C1(C(C)C)CN(C(C2CCC2)=O)CCCN1C(c1nc(Cl)cs1)=O N1(C(C2(OC)CCOC2)=O)CCC(CCCNC(C2CCOC2)=O)CC1 C1(COC)(NC(C2OCCC2C)=O)CCN(C(c2sccc2S(C)(=O)=O)=O)C1 C1(C(=O)NCCCN(C(C2C(CCC)CCC2)=O)CC)CC(F)C(=O)N1 Cc1nnc2n1CCC(C(=O)N(C(C)CCNC(=O)C(=O)NC1CC1)C)C2 c1(CC(C)NC(=O)C(=O)NCC2CS(=O)(=O)CCO2)nc2ccccc2[nH]1 CC1CCOC(C(=O)N(C(C)(C(=O)NCCc2cnc[nH]2)C2CC2)C)C1 C1(CC=C)(C(=O)N(CC(O)COC)C)CCN(C(=O)CCOCC(C)C)C1 n1(CC)cc2ccc(C(=O)NCC(C)NC(c3cncc4ccsc34)=O)cc2n1 c1(C(N2CCC(OCC=C)C2)C(=O)NCCCSCC)cc2ccsc2n1C C1(CC(=O)NCC(CCC)C)CN(C(c2cccc(CC#N)c2)=O)CC12CC2 CC(C)C(O)C(=O)N1CC(CC(C)(C)CNC(c2ccn(C)c2)=O)C1 Cc1cc(-n2ccc(C(=O)NCCC(C)(C)O)n2)ccc1Cl CC1(C)CCC(CC(=O)NC2(c3cn(CCCC(=O)O)nn3)CCC2)O1 N1(C(C(C2CCOCC2)OC)=O)CCN(C(=O)CCCN=[N+]=[N-])C(C2CCC2)C1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(CCNC(c1csc(C(F)(F)F)n1)=O)CC C12(CC)CN(C(C3(SC)CC3)=O)C(CNC(=O)CC3CCCC(C)O3)(C1)C2 CN1C(=O)CSC1=NC(=O)c1cccc(=O)n1CC(=O)Nc1cccc(I)c1 c1(C(=O)NC(CC)CNC(=O)C(C)CC2CC2)noc2cc(F)ccc12 c1(C(=O)NC(CC)CN(C(=O)CCc2ccoc2)CC)cccc(Cl)c1O N1(C(CSCC(C)C)=O)CC2CCCC(C1)N2C(=O)CCNc1ccccc1Cl CCCC(C(=O)NC(Cn1ccnn1)C(=O)NCCCCS(C)=O)OC c1(C(=O)OCc2cc(C)c(Br)s2)cn2c(n1)CCCC2C N1(Cc2c(C)noc2C)CCc2c(ccnc2Cl)C1 N1(C(c2occ(C)c2)=O)CCN(C(=O)C(C2(O)CCCC2)F)CC1C(C)C C1(NC(CCCC(C)O)=O)CC2CN(C(c3ccc(NC=O)cc3)=O)CC2C1 C(=O)(CC(C)CC(C)C)NCC12OCC(NC(C(C)OCCCC)=O)(C1)C2 C#Cc1cccc(CC(=O)NCC(C(C)C)NC(=O)CC2CSCCS2)c1 c1(C(=O)NCC(C)NC(C(C(C)C)CN(C)C)=O)c[nH]c2ncc(Br)cc12 Cn1nc2c(c1C(=O)NC1CCCCC1NC(c1ccc(=N)[nH]n1)=O)CCC2 N1(C(C(CC)COC)=O)CC(F)(F)CC1(C)CNC(=O)CCCc1ccc(C)s1 c1(CC(=O)NCC2(NC(C3CC3F)=O)CCC2)ccccc1Br c1(OC)cc(C(=O)NC2CN(C(C3CCCC3)=O)C2)cc(Br)c1NC(C)=O c1(C(N(CCCNC(C2(C)CCCN2C)=O)C)=O)cnc(S(C)(=O)=O)s1 c1(C(=O)NC(CNC(C(C)N2CCCC2)=O)(C)C2CC2)cc(C(N)=O)co1 c1(C(=O)NCC(CNC(C(C)NC(c2ccoc2)=O)=O)F)cc(Cl)cnn1 C1(CNC(c2cc(C(C)C)no2)=O)CC(NC(c2cn[nH]c2)=O)C1(C)C C(=O)(C1Cc2ccc(F)cc21)N1CCN(C(CN(C)CC)=O)CC12CCC2 C1(C#CC(=O)N2CCC(C(C)(O)CNC(=O)Cc3cc(C)on3)CC2)(CC)CC1 C1(CC(=O)N(CC(=O)NCCC)CCC)CC(C)(C)CN1 C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(CCF)CCC1CO c1(C(=O)NCC(CN(C(Cc2scc(C)c2)=O)C)O)cc2c(F)ccc(F)c2[nH]1 C1(NC(CCOc2ccc(C)cc2)=O)CCN(C(c2ncc(F)cn2)=O)CC1C C1(CC)CCC(C(=O)N(CCCCCNC(=O)CCCc2csc(=N)[nH]2)C)O1 C(=O)(C1CCc2c[nH]nc21)NCC(CC=C)C(=O)Nc1ccc(Cl)cc1C C1(NC(=O)CC2CC=CC2)CC(F)CN(C(c2cc(Cl)ccc2O)=O)C1 N1(C(C(CNC(N(C)CC)=O)F)=O)CC(O)CC(C)(C)C1 c1(NC(C23N(C(COC(CC)(C)C)=O)CCC2C3)=O)cnc(C)c(C)c1 N1(C(C)C(N2CC(O)(CCNC(=O)CCn3cnnn3)C2)=O)CCCCC1=O c1(C(=O)NCCC2(NC(COCC(c3ccccc3)C)=O)CC2)n[nH]c(C)c1Cl Cc1ccnc2c(C(=O)NCCC3CC(NC(C4CC45CC5(F)F)=O)C3)cnn12 c1(OC)cc(N(C)CCN(C)Cc2cc(Cl)no2)ncn1 CC1CCC(CNC(=O)C=C2CCC2)N(C(=O)CN(c2ccncc2)C)C1 c1(-n2c(C(C)C)nc(C3CC34CC4)n2)c2ccccc2nn1C CCCC(C(=O)OC)C(=O)N1CC(NC(c2cc(C(C)C)[nH]n2)=O)C(N=[N+]=[N-])C1 N1(CC(=O)NCC(C)N(C)C(C2CC(CC3CC3)C2)=O)CCCC1=O N1(C(C2ON=C(CC)C2)=O)CC(NC(=O)Cc2ccccc2)C2(CCCC2)C1 CN1CCOC(C(=O)N(CCCNC(C2CNC(=O)N2)=O)CC2CCCC2)C1 c1(CNCc2nc(-c3ccc(OCC)cc3)oc2C)cc(Br)cc(Cl)c1F CC(C)C(CNC(=O)CCCC1CC1C)C(=O)Nc1ccc(F)cc1O N1(C(=O)C=CC2CC2)CCC2(CCN(Cc3ccc(Cl)cc3F)C2)C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(CNC(c2cscc2Cl)=O)C1 C(c1ccc(C)cc1)=CCC(=O)NC(CCC(=O)N(CCNC(C)=O)C(C)C)C N1(C(CC2(CO)CN(C(CC3CCN(C)C3)=O)C2)=O)CCC(C(F)(F)F)C1(C)C C(CCC(C)C(=O)N(C)C)NC(c1n(CCC)nnn1)c1ncc(CC)s1 C1(C(C(C)C)NC(C2CN(C(C)=O)C2)=O)CCN(C(C2CCCSS2)=O)CC1 CCC(C)C(O)CNC(c1cc(CNC(c2cnc(Cl)s2)=O)[nH]n1)=O O=C(CCCC(F)(F)CO)NC1CCN(C(C2CCOCC2)=O)CCC1CO N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(c2cc(C)ns2)=O)C1 C1(NC(CSCC)=O)CC2CN(C(c3cc(CO)on3)=O)CCN2C1=O c1(C(=O)NCCCCN(C(CS(=O)(=O)NC)=O)C)cc(F)ccc1C(F)F c1(C(=O)NCC(C2CCCC2)NC(=O)CCc2nccs2)cc(Cl)ccn1 N1(C(c2c(C)[nH]cc2)=O)CCC(C2CC2NC(=O)C=Cc2ccccc2F)CC1 C1(NC(C(OC)OC)=O)CCN(c2ccccc2C(F)(F)F)C1=O c1(NC(=O)N(C2CCCC2)CCO)ccc2cnn(CCc3ccccc3)c2c1 N1(C(CC=C=C)=O)CC(NC(c2ccccc2OC(C)C)=O)CC2(CCC2)C1 C(=O)(C(O)CCC(C)C)N(CCCNC(=O)CC(C)(C)c1ccccc1)CC c1(C(N2CCC(NC(C(C)n3cnnn3)=O)C2C)=O)cccc2c1CCCCC2 c1(CNC(N2CCOCC2Cc2ccccc2I)=O)ccc(Br)cc1 C1(NC(C2(C=C)CCC2)=O)CCCCC1NC(=O)CCN(C(CC)CC)C C1(C)(C(N2CC(NC(CC(C)(C)OC)=O)C(F)C2)=O)COCC1(F)F C(N=c1nc2[nH][nH]cc-2c(O)n1)C1CCC(NC(Cn2ccc(C)cc2=O)=O)C1 N(C1CCc2cc(CNC(C3(C#N)CC(=O)C3)=O)ccc21)C(C1(C)CC1(Cl)Cl)=O C=CC1(C(=O)NCCC2(O)CN(C(c3ccc(CC)[nH]3)=O)C2)CCC1 N1(C(C(C=CC)O)=O)C2CCC1CC(NC(c1ccc(OC)c(C(C)C)c1)=O)C2 N1(C(CCCC#C)=O)CCCC2(CC(NC(=O)C=CC(=O)N(C)C)C2)C1 c1(C(=O)NC2CN(C(c3[nH]cc(CC)c3)=O)CC2C(F)F)cccc2[nH]ccc12 C1(CC)C(=O)N(C)CCN1C(C1CN(C(c2cccnn2)=O)CCC1(C)C)=O CCCCC(C)CCC(=O)N1CCC2CCCC12C(=O)NCCCOC(C)C N1(C(c2cn(CCC)nc2)=O)CCCC(NC(C2C=CC=CC=C2)=O)C1 c1(C(=O)NC(CN(C(c2cccc3nn[nH]c23)=O)CC)C)cc(Cl)c(F)cc1F C1(CNC(c2ncn(CCNC(c3cccc(F)c3)=O)c2)=O)CC2CCCC2C1 C#CCC(CC(=O)NCC1CC2(CC2)C(=O)O1)NC(c1cc(Cl)c[nH]1)=O CCC(C)(C#N)C(=O)NC(CC(=O)N(CC(C)C(C)C)C)C(C)OC N1(C(=O)CSCC2CCCO2)CCN(Cc2cn(-c3nccs3)nn2)CC1 c1(C(N2C(C)(CNC(C3C(C)(C)C3)=O)CCC2)=O)cc(Br)cnc1N c1(CC)[nH]nc(C(=O)NCCN(C(C2OCCO2)=O)C2CC2)c1[N+](=O)[O-] c1(C(=O)NCC(CO)NC(C2CCCN(CCC)C2)=O)cc(C)cc(F)c1N C1(C(C)NC(COCc2onc(NC)n2)=O)CN(C(c2csnc2C)=O)CCO1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(CCNC(=O)Cc2cccs2)CC1 C1(NC(C2C(=C)C2)=O)CCN(C(C2C(C=C(C)C)C2(C)C)=O)C12CCCC2 Cc1cc(=NCCCCC#N)[nH]c(=NCCOCCS(N)(=O)=O)[nH]1 c1(C(=O)NC2(CO)CN(C(COCc3cc(C)no3)=O)C2)cc(Cl)c(C)cn1 C1(NC(c2nn[nH]c2Cl)=O)CN(C(c2cnc3n2CCC3)=O)CCC1F C(=O)(C1=CCc2ccccc21)N1CC(N(C(C(CC(C)C)OC)=O)C)C(C)(C)C1 C(=O)(C(CO)C(C)(C)C)C(C1=CN2CCC1C2=O)=O.C1(NCC#C)CCCC1 Nc1nccnc1C(N1CCCCC1CC(N1CCC(CO)CC1)=O)=O N1(C(c2cc(OCC)no2)=O)CC(CC(=O)NOCCF)C(C)C1 C12(C)CN(CCC1O)C2=O.C(C)(C)(C)OC(=O)NCCNC(=O)OC Cc1cc(C(N2CCOC(CNC(=O)CN3CC=CC3)C2)=O)n2nc(C)cc2n1 N1(C(CNC(C(CC)C)=O)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 CC1CC=C(C(=O)N2CCC2CNC(=O)Cn2ccc(Br)n2)CC1 C1(NC(CSCC(C)C)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)CC1O C(C)(C)(CC(F)C(=O)NCC1(C(N)=O)CC1)NC(c1cncc(C)n1)=O C1(NC(COc2c(C)ccc(C)c2)=O)CC2CCC1N(C(C1CCSCC1)=O)C2 c1(OC)ccc(CC(=O)NCC2CC(NC(=O)CC=C(C)C)C2(C)C)c(F)c1 C12(CNC(CN(C(CN(C3CC3)CC)=O)C)=O)CCC(CC1)CC2 Cc1cc(C(C)C(=O)NCCCCN(C)C(C2C3CCC(F)(F)C23)=O)cc(F)c1 c1(CC(=O)NC2CCN(C(C=CC)=O)CC2O)nnc(O)c2ccccc12 Cc1cc(CCC(N2CCC(CNC(C3CCCN3C)=O)C(C)C2)=O)cc(C)c1 C1(C(=O)NC2CN(C(c3c[nH]c(=NCC)s3)=O)CC2(C)C)CCCC2C1C2(F)F N1(C(C(CC)COC)=O)CCCC(C)(C)C1C(=O)NC1CCC2CCC12 C12(COC(Cn3cc(-c4c(C)ccc(OC)c4)nn3)=O)CC=CCN1CCC2 N1(C(c2ccc(OC)c(-c3cn(CC(=O)O)nn3)c2)=O)CCC2(CCC(O)C2)C1 CCCCC(O)C(C)C(=O)NCC1CN(C(c2ccc(C)cc2F)=O)CCCO1 C1(NC(C=CC(C)C)=O)CCCCN(C(c2ccc(Cl)cc2Cl)=O)C1 C(=O)(C(C)(C)C1CCN(C(=O)CC2CC3(CC3)C2)C1)NC(C1(C)CCCO1)C c1(C(N(CC(C)NC(=O)CCCS(N)(=O)=O)C)=O)ccc2c(c1)OCCO2 Cc1ccnn1CC(N1CC(O)(CCNC(=O)CCSCc2ccccn2)C1)=O Cc1cc(C(N2CC3CC2C3C(=O)NCCc2ccccc2)=O)nc2nccn12 O=C(CCCCC(F)(F)F)NC1CCC2CCC1C2 C1(OC)CCCN(C)C1C.N1(C(C=CCOCCOC)=O)CC2(C1)CC(=O)N2 c1(C(N2CCC(CNC(CCC(=O)NC)=O)C2)=O)sc(C#N)cc1Cl C(CCCCCC(C)C)n1cc(C2N(C(CC(C)(C)OCC)=O)CCCC2)nn1 N1(C(Cn2ncc(C)c2)=O)CC2CCN(C(C3COCC3C(F)F)=O)CCC2C1 c1(OC)cc(N)c(Cl)cc1C(N1CC(NC(C2CC23CCOC3)=O)C1)=O c1(C(N(C2CCC(NC(=O)Cc3cccs3)C2)C)=O)cc2c(nc1O)CCCCC2 C1(NC(Cn2nc(C)c(Cl)c2C)=O)CC12CCC(NC(c1cccnn1)=O)CC2 n1(CC(N2CC(C(C)NC(C3(C(F)(F)F)CC3)=O)C2)=O)nnc(-c2ccco2)n1 C=CC(C)(CCOC)C(=O)NC(C)C(=O)NC(C)CCC1CC1 C(=O)(CC(C)(C(F)F)NC(N)=O)N(C1CCCN(C(=O)CC2=CCCCC2)C1)C C1(NC(C(C)OCC2CCCO2)=O)CN(C(c2c(F)cncc2Cl)=O)CCC1F c1(N(C(C)=O)C)ccccc1C(=O)NC(C)C(C)NC(C1(C)CC=CCO1)=O N1(C(C(=O)NCC2CN(C)CC(C)O2)=O)CC(c2ccccc2)C2CCCC12 c1(-c2nn(C(CC)C)c(C(F)(F)F)c2)ccc(C(=O)O)cc1F C(c1ccc(C)cc1)=C(C(=O)NC(CN(C(c1ccc(CC)nc1)=O)CC)C)C CCCC(C)(O)C(=O)N(CCCCN(C)C(C1(C)CCN(C(C)=O)C1)=O)C CC1CC(NC(=O)C(c2ccoc2)NC(c2c[nH]c(=N)o2)=O)CC(C)C1 C1(NC(c2cc(NC(=O)OC(C)(C)C)no2)=O)CCOC2(CCS(=O)(=O)CC2)C1 C1(NC(C2C(C)C2)=O)CN(C(=O)C=Cc2cncn2C)CCC1CO C(=O)(CC(C(C)(C)C)NC(=O)CC1(CSC)CC1)NC1(CCC)CC(C)(C)C1 CCN=c1[nH]c(C(N2CC(NC(c3cccc(F)c3F)=O)C3CC23)=O)cs1 Cc1ncc(C(=O)NCC2CCN(C)C2)c(Cl)c1Br c1(C(=O)NCCOCCCNC(C(CCSC)O)=O)ccc(S(C)=O)cc1 C1(C)(NC(C)=O)CCN(C(=O)C(N2CCOCC2c2nc(C)no2)=O)C1 N1(C(Cc2c(C)noc2)=O)CC(NC(=O)C=Cc2cscn2)C(O)C1 c1(-c2cn(CCCCCCC(C(C)=CC)=O)nn2)ccc(F)c(S(C)(=O)=O)c1 CC1CC(NC(C2CC(C#N)C2)=O)CCN1C(=O)COc1c(Cl)cccc1Cl N1(C(C(C)(C2CC2)OC)=O)CCCC(CCNC(C2CC(C3CC3)=NO2)=O)CC1 CC1(C(=O)NCC2(O)CC(NC(=O)CN3CCCC3CO)C2)CC=CCC1 c1(C(N2CC(CNC(c3cc(Cl)ccc3Cl)=O)C(O)C2)=O)ccn2ccccc12 c1(C(=O)NCC(C2CC2)NC(C#CC2(C)CC2)=O)ncn2cc(Cl)ccc12 c1(-c2ccc(CN3CC(C(=O)OC)N(C)CC3)s2)nccn2cccc12 C1(n2c(CC)cnn2)NC(=S)N(C(C)CC)C2=C1C(=O)OC2 c1(C(=O)NC(C=CC(=O)NC(c2ccco2)CO)C)ccc(F)c(CO)c1 C1(CN(C)C)CCCN1C(=O)C(C1(O)CN(C(C2(Br)CC2(C)C)=O)C1)F C1(CNC(c2c(N)cn(C)n2)=O)CN(C(=O)CCCC(F)F)CC12CC2 CCC(C(=O)N1CCOCC1CNC(c1c[nH]nc1C(C)(F)F)=O)C(C)C N1(C(c2cc(OC)sn2)=O)CC(CC(N2CCC3C(C(N)=O)C3C2)=O)C2(CC2)C1 c1(N(CC(=O)NC)C)nccc(=NC(C)c2nc(O)n[nH]2)[nH]1 N1(C(CC2CCC(C)O2)=O)CC2CCC(C1)N2C(c1ccc(C(N)=O)o1)=O N1(C(c2c(Cl)cc(C)c(C)c2)=O)Cc2ccccc2CC1CNC(=O)CC(C)F Cc1c(O)ccc(C(=O)NCC2CCN(C(c3ccc(Cl)nc3)=O)C2)c1C C1(CNC(C(Cc2ccccc2)OC)=O)CC2CCC1N(C(c1ccsn1)=O)C2 N1(C(C(C(C)C)NC(c2ccc(Cl)cc2)=O)=O)CCC(O)CC(C)(C)C1 CP(C)(=O)CC(=O)NC(CC1CC1)CC(=O)N1CC2CC1C2 N1(C(CNC(CCCCC)=O)=O)CCCCC(NC(=O)C(=O)Nc2ncc[nH]2)C1 C(CC(=O)NCc1nc(C)co1)(C(F)F)NC(C1CCC(NC(C)=O)CC1)=O C1(N(C(CN(C(C2(C(=O)OCC)CC2)=O)CC)=O)C)CN(C)CCO1 C1(C(=O)NC2CCC(CN(C(C(CC)(F)F)=O)C)CC2)CCc2nccn2CC1 Cc1cc(C(=O)N(C)CCOCCCN(C(=O)C(F)n2cccn2)C)ccn1 c12ccc(cc1)C(=O)OC2.C1(CCNC(CC)=O)CC=CCC1 C1(NC(C2CC(CCC)C2)=O)CCC(NC(C2CC3C=CC2O3)=O)CC1 C1(NC(COC2(C)CCC2)=O)CS(=O)(=O)CC1NC(=O)C=CC1CCOCC1 N1(C(CC2ON=C(C)C2)=O)CC(C)CC1C(=O)NC(c1cccnc1F)C CN1CCC(C(=O)NCCCn2cccn2)(NC(=O)C(F)=CC2CC2)C1 C#Cc1cc(C(=O)NCC2(CC(=O)N)CC23CCC3)cc(N)c1.C(C(C)(C)C)=CC C1(N(CCCO)C(C2C3CN(C(C)=O)CC32)=O)CCCCC1(C)C N1(C(C2(C)C=CCC2)=O)CCC(C(F)CNC(c2cc(Cl)no2)=O)CC1 C(=O)(CCC(=O)NCc1cc(C(N2CCC(OCC(N)=O)C2)=O)n[nH]1)NC c1(OC)cc(Br)ccc1CNCCCCCN N1(C(C(C=C)O)=O)CCCC2CN(C(c3[nH]nnc3COC)=O)CCC12 C1(NC(CC=C=C)=O)CC(OC)CN(C(=O)CN(c2ncccn2)CC)C1 c1(NC(C2C(NCc3c(C)n[nH]c3)C2)=O)ccc(I)c(CO)c1 C1(C(=O)OC)CC1C(=O)N(CCCF)C.C1C(=O)NCCN1C Cc1cc(CNC(C2CCCN2C(=O)CN2CCCCC2C)=O)nc(N(C)C)n1 c1(C(=O)NCCNCC2CC=CCC2)cn(CCOC(C)C)nn1.C1CO1 c1(C(=O)NC2C(CNC(c3cn(C)nn3)=O)C2)ccnc(-n2cncn2)c1 C1(C(=O)NC2C(C(=O)NCCCCC#N)CCC2)CCNC(=O)C1 c1(C(=O)OC)nc(N2CCC(CNC3CC4C=CC3C4)C2)ncc1Cl N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2C(CCN2Cc2ncc[nH]2)C1 C1(C(N2CC(CNC(c3n(C=C)nnc3)=O)C2)=O)CCn2c(cnc2C)C1 CC1(C)Cc2cccc(CNC(=O)NCC34CCCC(C)(C3)OC4)c2O1 N1(C(=O)OCC)CCC(C)(C(N2CCC(CSC)C2)=O)C1 c1(C(N2CC(NC(c3n(CCCC)ncc3)=O)C(C)C2)=O)cc(F)cc(C)c1N CCCCC(=O)C(=O)N(CC(C)NC(=O)CCN(C(=O)COC)C)C(C)C Cc1cc(C(=O)NC2CCC2CNC(=O)CNC=O)c2ccc(Br)cc2n1 c1(CSCC(=O)NC(CNC(C2C(C)(C(=O)OCC)C2)=O)CO)ccc(F)cc1 CC1CCN(C(C23CC(C2)S(=O)(=O)C3)=O)CC1NC(c1cccc(=S)n1O)=O C1(CNC(=O)C=CCF)CC2COCC2N1C(=O)C(O)CC1CCCCC1 N1(C(C2C(C)C2)=O)CCN(C(=O)C(c2cc(Cl)ccc2Cl)(C)C)CC1CCO N(C1CN(C(=O)CCCC2CC2)Cc2ccccc21)C(CC1C(=O)NCCC1)=O c1(CC)cccnc1C(=O)NCCCC1CCCN1C(=O)CN1CCCC1=O Cc1cn2c(CCC(=O)N(CC(C)NC(C3CC4(CC4)CO3)=O)C)csc2n1 CCS(=O)(=O)CC(=O)NCCCCCN(C(=O)C(C)(C)C1CCCO1)C c1(C(N2CCOC(Cc3cn(C4CCOCC4O)nn3)C2)=O)cccc2cncn12 CC1=NOC2(C1)CN(C(=O)NCc1nc(-c3ccc(F)cc3)oc1C)C2 c1(NC(C23CCC(C2)NC3)=O)nccc(Br)c1Br CC1CN2CCN1C(C(=O)NCC1CCN(C(=O)CCCC(N)=O)C1)C2 N1(C(c2c(Cl)ncc(C#N)c2)=O)CCC2(CCCC2N2C3COCC2C3)CC1 c1(C(=O)NC2CN(C(C3C(C(C)C)CCO3)=O)CC(C)C2)c(F)cc(F)cc1F C1(SC)CCN(C(c2nc(C)co2)C(=O)NCC2CCOC2)CC1 C1(CNC(C(CCC)NC(C)=O)=O)(CO)CC12CCN(C(=O)C(C)NC=O)CC2 C1(NC(c2cc(C)ncn2)=O)CC2CCC1(NC(=O)CC1(N(C)C)CCC1)C2 Cc1ccc(C(F)(F)F)cc1Nc1cn(C(c2ccccc2)C(N)=O)nn1 N1(C(C2(c3cc(C)on3)CC2)=O)CCN(C(C2CC3CCCC3C2)=O)CC1CO CCCC(C)C(=O)NCC1(CNC(=O)C(F)CN(CC)CC)CCOCC1 C1(C(N(C(C(N)=O)C2CC2)C)=O)CN(C(c2ccc(CO)cc2)=O)CCO1 O=C(N=c1ccn(C2CCSCC2)[nH]1)c1ccc(O)c(Cl)c1 C1(NC(C(C)CC(F)F)=O)CN(C(=O)Cc2cc(Br)cs2)C2(CCC2)C1 Cc1cc(C)c(C(=O)NC2CC(N(C(=O)C3=NNC(=O)C3)C)C2)c(S)n1 C#Cc1cc(F)c(C(N2CCC(NC(=O)C=CSC)C2C)=O)cc1F N1(C(C2N(N=O)CCC2)=O)CCC2CCC(C1)N2C(c1cc2cccnn2n1)=O CC(C)(C)CCC(F)C(=O)NCCSCO.N1Cc2cc(F)cnc2C1 N1(C(C(=O)NCC2CC2)=O)CC(CNC(c2ccccc2F)=O)N2CCC1C2 C1(C(=O)NCC#CCC)CCCCCCN1C(c1ncc2ccccn12)=O c1(CCCC(=O)NC2CCCN(C(c3ncn(C)c3)=O)C2)ccc(C#N)cc1 c1(C(=O)NC(CC=C)CNC(c2[nH]cnc2C)=O)nc(Br)n2ccccc12 N1(C(C(N2CC(C)OCC2)=O)=O)CCCC2CCC(C)CC12 c1(CNC(C2CCC(n3cc(-c4cc(C)on4)nn3)C2)=O)cc2oc(Br)cc2[nH]1 c1(C(N(C)CC2CCN(C(c3cc(Cl)on3)=O)C2)=O)cc2ccc(F)cc2s1 c1(CNC(C2CC=CCO2)=O)ccc2c(c1)CN(C(=O)CCC1OCCO1)C2 C1(NC(C(CCOC)C)=O)CCN(C(c2cnc(-c3ccsc3)s2)=O)CC1(C)C Cc1ncncc1C(=O)NCC1CCC(C(N2CC3CC2CS3)=O)O1 C1(c2cn(C3CN(C(=O)OC(C)(C)C)CC3F)nn2)COC(C)(C)OC1 c1(C(=O)Nc2ccc(NCc3cc(C(=O)OC)[nH]c3)nc2)ccc(Cl)c(F)c1 CCC(C)(C)C(O)C(=O)N1CCC(C)C(NC(c2cc(C(N)=O)c[nH]2)=O)C1C Cc1cn2cc(CC(=O)NC3COCC3NC(C3(Cl)CC3(C)C)=O)nc2s1 C(C(C)(C)C(=O)NCCN1CCC1)N(C)C(c1cc(=N)[nH][nH]1)=O c1(CC(=O)NC(CNC(C=CC(C)C)=O)CO)ccc(S(=O)(=O)N(C)C)cc1 CC1CCCN(C(=O)C(=O)N(CCCCNC(C2CCCN2N=O)=O)C)C1 N1(C(c2c[nH]c(=N)s2)=O)CCC(NC(c2ncccc2Cl)=O)C(CO)CC1 C1(CNC(COCCCCC)=O)CCCN(C(c2[nH]c(C)nc2C)=O)CC1 C(=O)(CC(C)CC(C)C)N1CCC(NC(c2c(CC)ocn2)=O)C(CO)C1 C12(CNC(=O)CCn3cnnn3)CCCC(CN1C(c1cccc(F)c1)=O)C2 c1(C(C)C)ccc(CC(=O)NCC2CN(C(=O)CCCC3CCC3)CC2O)cc1 C(=O)(C1Cc2ccc(F)cc21)NC(CC)CNC(c1ccc(C)n(C)c1=O)=O c1(NC(C(C)NC(=O)NC2(C#C)CC2)=O)ccc(S(N)(=O)=O)cc1 c1(C(=O)NC(COC)C)ncn2cc(-c3ccc(SC)cc3)sc12 Cc1ncc(Br)cc1NC(=O)C(O)C(F)F C(=O)(C(=O)N=S(C)(C)=O)N1CC(N(C(c2c(CC)nc(C)nc2)=O)C)C(O)CC1 CCCCC(C)C(=O)N1CCC(C(=O)NCc2nnc(C)s2)(CO)C1 C(=O)(C(C)(O)CCC)N(C(CC(=O)NC(CCC)CCC)(C)C)C Cc1c[nH]c(C(=O)NC2(C)CN(C(c3ccn(C)n3)=O)C2)c1 c1(N(C(=O)C2CC2)CC2CCCN2C(=O)C=CCBr)cccc(-c2cccnc2)c1 C1(C(=O)NC2CN(C(c3cncnc3)=O)C3CC23)CCCCCCC1 c1(OC)ccc2c(c1)c(CNC(=O)C(=O)NCC(F)F)c(C)n2CC(C)(C)OC C1(C(=O)NCCCN(C(=O)C=Cc2cscn2)C)CCCC1(C)O c1(CC(=O)NCCN(CC(C)O)C(c2cnns2)=O)nccn1C CCS(=O)CC(=O)NC1CN(C(=O)Cc2c[nH]nc2O)CC1C C(N=c1[nH]c(N2CCC(c3nncs3)C2)nc2c1SCC2)c1cccc(CC)n1 C(C(C)(C(C)C)NC(C1CCN(C(C)=O)C1)=O)NC(C(C)(C)OC)=O C(=O)(C(C)(CSC)NC(=O)CC1OCCC1(C)C)NC(CC)CCOC.OCC C1(NC(c2c(C#C)c[nH]n2)=O)CC1C1CCN(C(=O)CCOCCCOC)CC1 Cn1nc(C(N2CCC(CCC(=O)N3CC(n4cccn4)C3)C2)=O)cc1O N1(C(C2C(OCC)C2C)=O)CC2CCN(C(=O)Nc3c(C)cc(C)nc3C)C2C1 C1(c2nnnn2CC2CCOC2)(NCC(=CC(=O)NC)C)CC1C(C)C c1(N2C(CNC(C(C)=C(C)C)=O)C(C)CC2)ccc2c(n1)CC(C)(C)CC2=O N1(C(CCCCOCC)=O)CCC(NC(=O)CCSCC(C)C)C(F)C1 C1(NC(CSCCCC)=O)COCCN(C(=O)CCC2COC(C)(C)O2)C1 N1(C(C#CC)=O)CCC(C(=O)OCc2ccc(C)c(-c3ccccc3)c2)C(F)C1 c1(NC2(C)CC(NC(C3CC(F)(F)C3)=O)C2)nc(C2CC2)nc2[nH]ccc12 C=CCC(CC)C(=O)NCC1(O)CN(C(c2ccc(C(F)(F)C(F)F)cc2)=O)C1 N1(C(C(CC)C)=O)CC(CNC(c2cn(CCC3CC3)nn2)=O)C(O)C1 C1(CNC(Cc2ccc(OC)s2)=O)CC(C)(C)CN1C(c1nn(C)c(Cl)c1Cl)=O C1(C2N(Cc3cn(CC(=O)OC)nc3)CCC2)CCC(C)CC1 CC1CN(C(c2cnsc2)=O)CCCN1C(=O)CC(=O)Nc1nccs1 Cn1cc(Br)c(CS(N2CC(C(=O)O)C(C(F)(F)F)C2)(=O)=O)n1 CC1CCCC(CC(N2CCCC2C2(C(=O)NCCC(=O)N(C)C)CC2)=O)C1 CN1CCn2cc(C(N3CCOC(CNC(=O)CCP(C)(C)=O)C3)=O)nc2C1=O N1(CC)C(=O)CCC1CC(=O)NCC(CO)NC(c1n[nH]cc1OC)=O c1(-c2n(-c3n(C)c(Cl)nc3Cl)ccn2)cc2ccccc2n1CC(=O)O c1(C(N2C(C(C)C)C(NC(=O)CCC#N)CC2)=O)nc(Br)c2n1CCCC2 N1(C(C(CCC)C)=O)CCOC(C)(CNC(=O)Cc2c(C)cccc2C)C1 Cn1cc(C(=O)NCC(CNC(C2(n3nccn3)CC2)=O)CO)n(C)c1=O C1(COC)(CNC(C2CC(CF)C2)=O)CCCN1C(=O)CCc1c(C)noc1C C1(C(N2CC(C)C(CNC(=O)C3=COCCO3)C2)=O)CCc2ncnn2C1 n1(CC)c(C(N2CC(C(C(=O)NCC3(CCO)CC3)OC)C2)=O)cnc1O CCCS(=O)(=O)C(C)C(=O)N(CCCCN(C(=O)C1=C(C#N)CCC1)C)C c1(C(N2CCCC(C)(C(=O)Nc3ncc(C(C)=O)s3)C2)=O)cn2c(Cl)cccc2n1 N1(C(CSCC=C)=O)C(C)CN(C(=O)Cc2occc2C)CC1C C1(C(=O)NCC2(C)CCCO2)CC(O)CN1C(=O)CSc1ccc(O)cc1 Cc1cc(C(=O)NCC2(F)CCN(C(C3CCCCCCC3)=O)CC2)nc(C)n1 c1(C(N2C3CC(NC(C4C(C=C)CC4)=O)CC2CC3)=O)cc2c(C)cccn2n1 C12(CNC(Cc3cc(C)no3)=O)CN(C(C3CCCCS3)=O)CC1CCO2 N1(C(C(C)S(N)(=O)=O)=O)CC2(CCCCN(C(c3ccnnc3S)=O)C2)C1 N1(C(C(C)(C)F)=O)CC(CC(=O)NC2C(O)CC2O)C2(CC2)C1 Cc1cccc(CCC(=O)NCCN(C(C2CCC23CCC3)=O)C2CC2)c1 C(C(CC(C)C)C(=O)N1CCOCC1C1CCC1)NC(c1cncc(C)n1)=O C1(CNC(CCOC)=O)CCC2(CCC2)C1NC(c1cccc(O)c1C)=O CCCC(O)C(=O)N1CCC1C(=O)NCCC(F)(F)CO C=CCC(C)(CC)C(=O)NCC(CO)NC(=O)CSC C1(CC)CCN(C(=O)CC2C=CC(NC(C3(CO)CC(C)(C)C3)=O)C2)CCO1 C1(C(=O)NCC(CC(=O)OC)O)CCC2CCC1N2C(=O)C(F)(F)C1CC1 C1(CNC(N2CCC(C3CCCCO3)CC2)=O)CC2CCC2C1 Cc1c(NC2(CO)CCOC2)ncnc1N1CCCC(C)C1 c1(N2CC3C(C(=O)Nc4cn(CCOC)nc4C)(C3)C2)ncc2[nH]ncc2n1 C(C(C)(C)CC(=O)N1CCC(CNC(=O)C(O)Cc2cnc[nH]2)C1(C)C)N(C)C N1(C(CCNC(=O)CO)=O)CCCC12CCN(C(c1ccoc1Cl)=O)C2 C1(C(=O)NCC2CN(CC)C(=O)O2)CC2CCC(C1)N2C(=O)CCC1CC1 CC(CC(=O)N1CCC1C(=O)NCCCc1nncn1C)C1CC1 NC(=O)CC(N=c1ccnc(NC2CC3CCCCN3C2)[nH]1)c1ccc(Cl)cc1 CC1C(NC(=O)Cn2cccnc2=O)C(C)CCN1C(=O)C(C)n1ccnc1 CC(C)CC(C1CC1)NC(C1CCCC1)CC1CCOCC1 c1(C(N2C(CC(=O)Nc3ccc(F)cc3)C3CCCC32)=O)cccc2[nH]ccc12 Cc1ccc2c(=NC(C)c3ccc(Br)cn3)[nH]c(=NCC(C)CO)[nH]c2c1 CC1CN(C)C(=O)CN1C(=O)C(CC(F)F)NC(=O)C=Cc1cnn(C)c1 N1(C(CCN(C(C2CC(C)(O)C2)=O)C2CC2)=O)CC2(COC(=O)C2)C1 C=CC(C)CC(=O)NC1CCC(N2CCN(C(C3COC3)=O)CC2)CC1 c1(SC)nc(=NCc2cscn2)s[nH]1.c12ccccc1CO2 C1(C(N(C(C)C)CC)=O)CC(NC(=O)C(C)NC(C2CCC2)=O)C1 c1(OC)cccc(CN2CCCC(C(=O)NCC3CCO3)C2)c1C C1(CC)(NC(=O)CC(C)C(C)C)CCCN(C(c2ccncc2OC)=O)C1 C(CC)(CCC(=O)N(CC(O)CF)C)NC(c1[nH]cc(C(C)=O)c1)=O N1(C(C(C(C)C)OC)=O)CCC2(CCN(C(c3ccc(F)nc3)=O)C2)C1 N1(C(C2(C)CCNC2=O)=O)CC2(C1)CN(C(=O)C=Cc1cn[nH]c1)CCO2 c1(C(N2CCN(C(C3CCCCC3)=O)C3CC23)=O)ccc2c(O)nnc(O)c2c1 c1(NC(N2CCC(N3C(=O)CCC3=O)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(C(=O)N1CCN(CCCNC(C23CC(CCO2)C3)=O)CC1)C(C)C C1(C(N2C(CNC(Cn3c(C)ncc3)=O)CCC2)=O)CC2C=CC1C2 C1(NC(CCCCC)=O)CC2(CCCN(C(=O)CNC(=O)CC3CCCC3)C2)C1 Cc1cc(C(N2CCC(C(C)NC(C3CCSC3)=O)C2)=O)nn1C(C)(C)C CC1CCN(C(=O)C=C2CCC2)CC1NC(c1cnc(-c2cccnc2)s1)=O n1(CCC(=O)NC2CCC(CCNC(CSC)=O)C2)c(C)cc(O)cc1=O c1(COC(C2CC(=O)N(C3CCCC3)C2)=O)ccc(COc2ccccc2)nc1 CC(C)(Cc1cnn[nH]1)C(=O)NC(CNC(c1csc(=N)[nH]1)=O)CO C1(C2CN(C(=O)C(c3ccccc3)=O)C2)(NC(Cc2c(C)cc(C)s2)=O)CC1 N1(C(C(C)SCCCC)=O)CC(NC(=O)CC(C)CCC)C(C)(C)C1 c1(C(=O)NC(CNC(CC(=O)OC)=O)C(C)(C)C)cnc2ncnn2c1C C12(NC(C3(NC(C)=O)CCCC3)=O)CC(C1)N(C(c1scc(C)c1C)=O)C2 c1(C(N2C3CN(C(c4c(NC)nsn4)=O)CC2C3)=O)ccc2cncn2c1 C1(C(=O)NCCCC(C)NC(=O)CO)CC2(CCC2)C1 C(=O)(CC(C)C(=O)NCC(C)(F)CNC(C1CN(C)CCO1)=O)OC C1(CNC(=O)OC(CCNC(C2CC(C(=O)OC)C2)=O)=O)CCCOC1 N12C3CCC1C(C3)C2=O.c1(N(C(c2ccc(C)[nH]2)=O)CCO)cccc(Cl)c1C C1(OC)CN2CCCC2(C(=O)N(CC#N)CCCCN=c2nn[nH]n2C)C1 C(c1ccc(Cl)cc1)=CC(N1CCC(CCNC(C2(Cl)C(C)(C)C2)=O)C1)=O c1(C(=O)NC(C(N2CC(C(=O)OC)C2)=O)C2CCC2)n[nH]cc1[N+](=O)[O-] C#Cc1ccc(C(N2CC(NC(=O)C(C)(C)OC(C)C)C(F)C2)=O)c(C)c1 O=C(CC1CN(C(=O)CN(CCO)CCO)CCO1)N=c1cc[nH]c(C(F)(F)F)c1 C1(CCNC(=O)Cn2nccn2)CCCCN1C(c1ncncc1Cl)=O C(CCCCC(=O)N1C2CCC(C2)C1C(N1CCC(n2ccnc2)C1)=O)N(C)C N1(C(C2(CC)CC2)=O)CCC(NC(c2nc(C)nn2C)=O)C(CC2CC2)C1 c1(C(=O)NC(CC)CNC(C2CC2C)=O)cc2cc(OC)ccc2nc1C c1(C(=O)NCC(C)(CC)NC(C2CC2CC(=O)OC(C)(C)C)=O)ccc(F)c(Cl)c1 C1(NC(C2CCC(F)CC2)=O)C=CCN(C(=O)C=Cc2ccccn2)C1 c1(NC(=O)C(c2ccccn2)O)ccc2c(c1)CN(C(C1(F)CCCNC1)=O)C2 c1(C(=O)NCCN(CCC)C(C2(F)CCOC2C)=O)cc(C)nn1C(C)(C)C c1(CCNC(C2(C)CSC2)=O)ccc(CNC(=O)CC2CCC(=O)N2)cc1 C1(C(=O)OC(C)(C)C)CCc2nncn2CC1.C1(OC)CC(C(=O)O)N(C=O)C1 c1(C(N2CC(CC)N(C(c3cnncc3O)=O)CC2)=O)cnc2sc(C)c(C)n12 CC(C)(C(=O)N1CCC1CNC(c1ccc(-c2ccccc2)[nH]1)=O)C1CCCCC1 C(=O)(CCN=c1cc(C)[nH]c(=NCC2CC3CCC(C2)S3)[nH]1)NCC C1(C(=O)NC(CC#C)C(=O)NCC2CC3(CCC3)CO2)CC(C)(C)CCO1 C1(C(=O)NCCCN(C(=O)CSc2ccncc2)C)CC2(CCC2)CO1 C=CCC(C(=O)N1CCC(F)(CNC(c2cncnc2CC)=O)C1)OC C(N=c1nc(N2CC3CN(C)CC3(C)C2)c2c([nH]1)CCCCC2)c1c(C)ocn1 N1(C(CN(C2CC2)CC)=O)CCC(NC(c2c(C(F)F)cccc2F)=O)C1(C)C c1(C(=O)NCC(CNC(CC(C)(C)OC)=O)O)cnc2cc(Br)ccn12 C(C(C)(C)CCNC(=O)C=C(C)C1CC1)NC(CCN(C(CCC)C)C)=O c1(CCCNC(C23COCC2CN(Cc2ccoc2)C3)=O)ccccc1[N+](=O)[O-] CC1(C)CCCC(C(N2CC3CC2C3C(=O)NC2CC3CCC(C2)S3)=O)C1 c1(C(=O)NC2C(CNC(C(C=C)(C)CC)=O)COC2)c[nH]c2c(Br)cccc12 c1(OC)c(Br)cc(NC(c2ccc(-c3cscn3)cc2)=O)cc1Br C1(C(N(CCCCCO)C)=O)CC12CN(C(C1CC(O)CN1)=O)C2 CC1C(C)N(C(c2ccco2)=O)CCN1C(=O)CNC(=O)OC1CCC1 C1(C)(CCNC(CCOC)=O)CCN(C(=O)C(C)Cc2ccc(N)cc2)C1 c1(C(N2CCC(N(C)C(c3coc(O)n3)=O)C2)=O)cccc(C2CC2(F)F)c1 C1(CCOC)(NC(C2CCC3(CC3)C2)=O)CCN(C(=O)CCOCC2CC2)C1 C1(NC(Cn2c(C)ncc2)=O)CC(NC(=O)CC(C)C2CCCCC2)C(O)C1 c1(OC)cccc(-n2cc(CC3CCCN3CC3CC(F)(F)C3)nn2)n1 C1(C(=O)NCC(CC=C)(C)C)CN(C(=O)C(CCC)OC)CC1(F)F C1(NC(C(C)CN2CCOCC2)=O)CCN(c2nnc(C(F)(F)F)s2)C12CCC2 Cc1ncc2n1CC(NC(c1c(Cl)sc(N)c1C)=O)CC2 CC1(C)CCC=C(C(=O)NCC2CC(F)(F)CN2C(=O)CCc2nc[nH]n2)C1 C12(CNC(C(c3ccc(C)cc3)C)=O)CCCC(CN1C(c1cnsn1)=O)C2 C1(CNCC2C(C)(C)CO2)CCN(C(=O)C(c2ccccc2F)O)CC1 C1(C(N2CC(C3OCCN(C(=O)CC4CC4C4CC4)C3)C2)=O)CN2CCC1CC2 C(CC(C(=O)N1CCC1CNc1cccs1)NC(c1cc(Br)cs1)=O)SC N1(C(CCC#CC)=O)CC2(CC(CNC(c3cccc(NC4CC4)c3)=O)C2)C1 C1(CC=C)(NC(C2CCN2CC2CC2)=O)CCCN(C(=O)CN(C)C)C1 C1(CNC(C2(CNC(c3cc(F)ccc3O)=O)CC23CCC3)=O)CC2(CCO1)CC2 C=Cc1ccc(CN(C=O)CC(=O)N(C)C(c2c[nH]ccc2=O)C)cc1 C1CC(C)(C)NC(=O)C(C)N1C.c1(C(=O)NC2CC2CO)cc(C2(C)CC2)on1.CCO C(CCCCCNC(C1CCCCC1)=O)N(C)C(c1ccc(C2CCOC2)s1)=O c1(C(=O)NC2CN(C(c3ccc(C)c(O)n3)=O)CC2CO)cc2cccn2cn1 C1(C(N(C)CCc2nccs2)=O)CCCCN(C(=O)CCCF)C1 C12(C(N3CC(COC)(CNC(C4CSCCS4)=O)C3)=O)CCCC1CC(=O)CC2 C#Cc1cc(C(N2CCC(NC(=O)COCCCF)C(C)C2)=O)cc(Br)c1 Cc1cc2ccc(C(=O)NC3CCOC3C3CC3)cn2c1 c1(OC)cc(OC)nc(C(N2CCC3CCC23CNC(=O)C2=COCCC2)=O)n1 c1(C(=O)NC(CNC(CCC)=O)C2CCC2)ccn2ccnc2c1 CC1CC2(CC(C(=O)NCCCCC(=O)N3CCOC(C(C)C)C3)C2)C1 C(C)(C)(C(C)CC(=O)NCc1cn(C(C)C)nn1)NC(CCC(C)=O)=O CC(C)CCC(O)C(=O)N1CCCC(CC(=O)NC2C(O)CC2O)C1 c1(N2CCC(C(N(c3cncc(F)c3C)CCC)=O)C2)ncc(NC)cc1Cl N1(C(C2C(OC)CC2)=O)CCC(CF)(NC(c2ccccc2NC2CC2)=O)C1 N1(C(C2C3N(C(c4c[nH]c(=NC)o4)=O)C(CC3)C2)=O)CCCN(C)C(=O)C1 N1(C(C2C(C)(C)CC2)=O)CCn2c(CNC(C3(C)C=CCCC3)=O)nnc2C1 c1(OC)ccc(CN2CCC(C(N3CCCC3CO)=O)C(O)C2)c2ccccc12 c1(N(C)Cc2ccncc2Cl)cc(S(=O)(=O)NC(CO)CC(F)(F)F)ccc1C#N C1(CNC(c2ccc(C)n2C)=O)CN2CCCCC2CN1C(=O)COCC(F)F N1(C(c2nn(CC)c(C)c2)=O)CCC12CN(C(c1cc(CC(C)C)c[nH]1)=O)C2 C1(CCOC)CN(C(c2cnn(C3CC3(F)F)c2)=O)CCN1C(=O)CP(C)(C)=O c1(OCC)oc(C)nc1C(N1CC(CNC(=O)C=CC2(C)COC2)C(O)C1)=O C1(NC(C2N(C(C(CC3CCC3)OC)=O)CCC=C2)=O)CN(C)C2(CCC2)C1 c1(CC(=O)NCC(CNC(C2CC3C=CC2C3)=O)CO)ccccc1F c1(C(N2CCCC(NC(CC(=C=C)C)=O)C2)=O)cc(F)c(Br)c(F)c1 C#CCCC(C(=O)NC1CC12CC2)NC(C1CN(C)C1)=O c1(C(N2C(CCCC)CN(C(=O)C(C)O)CC2)=O)ccc(Cl)c(Cl)c1OC c1(OCC)cccc(NC(=O)C(CNC(c2cc(C)sc2N)=O)N(C)C)c1 c1(C(=O)NC)csc(COC)n1.C(=O)(C(C)C1CCCO1)C1(COCC)CC1 C(CC(C)C(=O)N1CC(F)(C(=O)Nc2cnn(CCF)c2)C1)=CC C(C)(CNC(c1c[nH]nc1-c1ccsc1)=O)(C(C)C)NC(Cc1c(C)nc[nH]1)=O C(CC(=O)NCCC(Cc1ccccc1)NC(C1CCC1)=O)(C(N)=O)NC(C)=O c1(C(=O)NCC#CCNC(CCc2ccc(C)s2)=O)cccc(C(F)F)c1C O=S(=O)(c1cccs1)N1CCC(n2cc(-c3cc(C4CC4)no3)nn2)C1 O=C(NOC(=O)CC1CCCCO1)C1=CC2(CCN(CC3CCCCC3)C2)C1 C=CC1(CC(=O)NC2CC(NC(=O)C(C)c3ccco3)C2)CCOCC1 Cc1ccccc1NC(C1CCC(CC(=O)NOCCOCCF)C1)=O Cc1ccc(CCNC(=O)C(=O)NC2C=CCCC2c2ccccc2)cn1 C1(C(N(CC(=C)C)C)=O)CC2CC1CC2NC(C1(CO)CCCCO1)=O C(CCC(=O)N1CCC(CN(c2cc(Oc3ccccc3)n[nH]2)C)C1)=CCC=C Cc1c(O)c(=O)ccn1CC(=O)NCC(C1CCCC1)NC(=O)C(C)n1ccnc1 C1(C(C2CCCN2C(=O)C(C)CC(=O)OC)NC(CCCC)CO)CC2C(C1)C2(F)F c1(C(N2C3CN(C(Cn4c(C)csc4=O)=O)C(C3)C2)=O)ccn2c1CSCC2 c1(NC2CCN(C(Cn3ccc(C)n3)=O)C(C)C2)ncnc2c1nnn2C(C)C c1(C(NC(=O)CC2CC(=O)NC2=O)Nc2scc(COC)c2)cccc(C#N)n1 CCCCCC(C)(C)C(=O)NCC(C)NC(=O)CCc1cccnc1F Cc1ccnc(C(N2CC3CC3(CNC(C3(C(F)(F)F)CCCCO3)=O)C2)=O)c1 C1(NC(C2(CSC)CCC2)=O)CCN(C(=O)CC2CCCOCC2)CC(O)C1 c1(C(N(C)CC2CCCN2C(=O)CCF)=O)cc2cccc(Br)c2[nH]1 CCC(CC(=O)N1CC(CCNC(c2sccc2CO)=O)(OC)C1)n1cccn1 N1(C(C2C(C)CCC2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)C2(CCC2)C1 Cc1ccc(NC(c2ccncc2)=O)cc1.N12CC(CC1C)C(=O)NOCC2=O c1(N(CC(C)(C)N)C(=O)CC2CCCOC2)ncc([N+](=O)[O-])cc1C.CO N1(C(c2cc(CNC(C=CCCC)=O)sn2)=O)CC(C2CC2)C1C1CC1 C(C(N)=O)(C(=O)O)NC(CONC(Cc1ccn(CCC)c1)=O)=O c1(C(CC)C(=O)NCCN(C(=O)CCCC)CC(C)O)cccc(C)c1 C1(C(N2C(CNC(CCN(CC(F)(F)F)C)=O)CC2)=O)CC(=O)NC(=O)N1 C1(NC(CC23CC(C)(OC2)C3)=O)CCC2CCN(C(c3c[nH]cc3Br)=O)C1C2 S(=O)(=O)(c1ccc(C)cc1C)NCCN(C1CCCCC1C)CC c1(CCC(=O)NCC2C3CC2N(C(=O)C=Cc2ccoc2)C3)ccc(F)cc1F N1(C(C2(SC)CC2)=O)CC(CNC(c2ccnn2CCN(C)C)=O)CC(C)(C)C1 c1(C(N2C(C(N3CC(C)OC(C)C3)=O)CC2)=O)cc(Br)c2cn[nH]c2c1 c12ccccc1CC2.N1(C(C(=O)NCC)=O)CCC(c2ccccc2)CC1 C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(CCC(=C)Cl)=O)(CC)CC1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCO3)=O)C2)ccccc1O N1(C(C(C)O)=O)CCC(NC(c2ccc(-c3ccccc3)cc2)=O)C(F)C1 C12CC(C1)NC(=O)CO2.C1(C(=O)NC(C(=O)OC)C2CCCO2)CC1(C)C(F)F c1(N2CCCC(CCC)CC2)nc2c(c(=NC(C)C3CC3)[nH]1)SCC2 C1(CNC(c2cccs2)=O)CC2CN(C(=O)Cc3cc(O)nc(O)n3)CC12 c1(C(=O)NC(CNC(c2cccc(SCC)c2)=O)C)ccc(C(F)(F)F)cc1N c1(CNC(C2C(C=C)OCC2)=O)ccc2c(c1)CCOC2.C12CCCCN1C2=O c1(C(N2C(CN(C(C(C)C3CCC3)=O)C)CCC2)=O)coc2c1CS(=O)(=O)C2 n1(CC)cc(Br)c(=NC(=O)N2CCCC2c2nnc(C)o2)[nH]1 N1(C(=O)NC2C(C(c3ccccc3Br)=O)CC2)CCCC(CCF)C1 C1(C(N2CC(C)CC(CC)C2)=O)CC2CCC1N2C(c1cc(COC)no1)=O N1(C(CSCCC)=O)CC2(CCC(NC(=O)COC(CCOCC)=O)O2)C1 C(C)(CCCCCO)NC(C1(C)CN(C(c2nc(C)oc2C)=O)C1)=O C(CN=c1[nH]c(=N)[nH]c(=NCCCN2CCCCC2C)[nH]1)c1nc(C)c(C)s1 C1(NC(c2cc(C(C)=O)sc2)=O)CC(NC(=O)CC2CS(=O)(=O)C2)C12CCC2 c1(C(N)=O)cccc(C(=O)NC2CC(NC(C3OC4CCC3C4)=O)C2)c1F c1(C(=O)NCC(CC=C)NC(=O)C(F)C2CCCC2)nn(C(C)C)nc1Br CCC(C#N)(CC)C(=O)N1CCCCC(CNC(=O)Cn2nc(C)n(C)c2=O)C1 N1(C(C2(NC(=O)COCC)CC2)=O)CC2CS(=O)(=O)CC2(COC(C)CC)C1 N1(C(Cc2ccn(CC)n2)=O)C2CCCC1CN(C(c1cc(C)cc(F)c1)=O)C2 Clc1cnc(NC2CCN(c3ccccc3)C2)c(I)c1 N1(C(C(=O)Nc2ccc(N(CCO)CC)cc2)CC2(C)CC2)CCN(C)CC1 c1(CC)cc(-c2nc(CC(C)CC)no2)cc(Cl)n1 C1(NC(C2(C)CC=CC2)=O)CCCCN(C(=O)CN2CCCC2=O)CC1 C(=O)(CCC(=O)NC1CCCN(C(=O)C(C2CC(F)(F)C2)O)C1)N(C(C)C)C CCC(CNC(C1CCN(C)C1)=O)(CC)NC(c1ccc(C(N)=O)nc1)=O N1(C(CSC)=O)CCC(C2CC2)(CNC(=O)C(C2CCOCC2)F)C1 c1(C(N2CCC(NC(Cc3c(C)non3)=O)CC2C)=O)cnn(C)c1S(N)(=O)=O CCC(CC)C(C(=O)N1CC(NC(=O)CP(C)(C)=O)CC(C)(C)C1)OC C=CC1CCCC(NC(=O)C(C)(CNC(=O)CCOC)CC)C1.C1(C)CC1 C1(C(N2CCC(CNC(=O)CC(O)CN(C)C)C2)=O)(OCC)CC(F)(F)C1 c1(CSCCC(=O)Nc2ncc(-c3ccccc3F)o2)ccccc1Br CCS(=O)(=O)CCn1c(N(CC(C)C)C)nnc1CSc1nccs1 C(CCCCN(C(=O)C(C)(O)C1CCOC1)C)NC(CN(CCC)C)=O Cc1cc(C(=O)NCC2N(C(=O)CS(N)(=O)=O)CCCC2(C)C)c(N)c(Cl)n1 c1(OC)cc(C(=O)NC2CCSC23CN(C(C2CC2(C)Br)=O)C3)cc(N)c1O C1(NC(C2CC(OC)C2)=O)CCN(C(=O)CCSC2CCCC2)C(C)C1 C#Cc1ccc(C(=O)NCC2(O)CCCN(C(=O)C(F)CCCCC)C2)cc1C C12(NC(CC)=O)CC(C)(C1)OC21CN(C(c2ccc3nc(=N)[nH]n3c2)=O)C1 n1(CC(=O)NC2C3CN(C(C4=CCCC4C)=O)C(C3)C2)ncn2cccc2c1=O O=C1CCc2cccc(C(N3CCOC(C(N4CCC5(C4)CC5(F)F)=O)C3)=O)c21 C1(N(C(CC(=C)C)=O)Cc2ccccc2C)CCCN(C(C2CC2)=O)C1 CN1CC2(CCN(C(C34CCC3CN(C(=O)CC3CCC(=O)CC3)C4)=O)C2)C1 c1(C(N2CC(=C(CNC(C(C)O)=O)F)C2)=O)sc(C2CC2)nc1-c1ccccc1 N1(C(CCc2cc(C)[nH]n2)=O)CCCC(NC(c2csc(Cl)c2Cl)=O)CC1 C12CN(N3CC4CCCCCC4C3)CC1n1cc2nn1.CC(C)(C)OC(=O)CO CC(C)C(O)C(=O)N(CCNC(C1CCCCN1S(C)(=O)=O)=O)C1CC1 c1(C(N(C(CNC(c2c(CC)nco2)=O)C)C)=O)cc2nc(C)[nH]c2cc1F N1(C(C(=O)NC(C2CCCNC2)C)=O)CCC(C(C)(C)C)CC1 c1(C(=O)NC(CCN(C(C(CC)=CC)=O)C)C)cc(Br)cc(C)c1F C1(COC)CCN(C(=NCCc2ccc(F)cc2)NCCc2nc(C)no2)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)C(F)C1CCC1)Nc1cnc(COC)nc1 c1(-c2c(C(=O)OC)n[nH]c2)cnc(C(=O)Nc2nc(CC)oc2)c(C)c1.CO c1(OC)ccc(C(C)C(=O)NC(C)CCNN2CCCCC2=O)cc1F N1(C(Cc2ccn(CC)n2)=O)CC2CN(OC(CC3(C(=O)OC)CC3)=O)CC2(C)C1 C1(OCC)CC2CN(CC(=O)NCCOc3ccc(Br)cn3)CCN2C1 C(CCC(=O)O)(C(=O)N1CC2CCC2(NCC2CCC2)C1)NC(=O)OC(C)(C)C n1(CC(C(=O)OCC)F)cc2ccc(NC(C3(O)CCOC3(C)C)=O)cc2n1 N1(C(C2(C(=O)NC)CC2)=O)CC(O)(CNC(c2ccc(-c3sccc3C)s2)=O)C1 O=S(=O)(c1ccc(Br)s1)N1CCCC(NCCOC2CCOCC2)C1 c1(C(=O)NC(CC)CNC(c2cnccn2)=O)ccc2c(C)cc(Cl)nc2c1 C1(COC)CN(C(C2OCCC2CNC(c2nonc2C)=O)=O)CCO1 c1(CC(=O)NCC(CN(C)C(C2CC2c2ccco2)=O)O)nc2c([nH]1)CCCC2 C1(C(=O)Nc2cnc(SC)nc2)CNC(=O)CN1C(=O)C(C)CCN(C)C C1(C(N2CC(C=C)C(NC(c3cncc(OC)n3)=O)C2)=O)CCCCC(C)(C)C1 n1(C(C)C)ncc(C(N2CCC(F)(CNC(C3(F)CC3)=O)C2)=O)c1Cl C1(C(=O)NCC2(NC(C3CC(O)(CC#C)C3)=O)CC(OC)C2)CCC2(CC2)CO1 c1(CNC(c2n(C(CC)C)nnn2)c2ncoc2CC)ccc(F)cc1 Cc1ccc(Cl)c(C(N2CCCC(NC(c3csc(-c4nc[nH]n4)n3)=O)C2)=O)c1 CCC(C)(C)C(O)C(=O)N1CC=CC1C(=O)NCc1cccc(OC)n1 C(=O)(NNC(=O)C(C)(C)CCCCNC(C1SCCC1C)=O)c1c(CC)ocn1 Cc1ncnc(C(N2CCN(C(c3cc(C4CC4)[nH]n3)=O)C(C(F)F)C2)=O)c1C c1(NC(C2CN(Cc3cccs3)CCO2)=O)ccc(I)c(Br)c1 C(=O)(C1Cc2ccccc21)NCCCCCNC(C(CNC(C)=O)(C)C)=O C(C1=CCN(C(c2ccc(C(C)C)o2)=O)CC1)NC(C(C)SC)=O Cc1ccc(F)c2oc(C(N3CCC(NC(=O)CC4CCC5CC45)C3)=O)cc12 c1(C(=O)NCCn2cc(C(N3CC=CC3)=O)nn2)ccc(O)cc1 C=CC(C)C(C)C(=O)NCC(c1ccc(F)cc1)NC(=O)C1=CC(C)(C)C1 c1(NC(CCCN(C(=O)OC)C)=O)cc(C)cnc1O.C(CCC(=O)N)C1CCC1 C12(NC(CCNC(=O)C3CC3)=O)CCCC1CN(C(C1CCCCC(=O)N1)=O)C2 c1(NCc2c(C(C)(C)C)noc2)[nH]c(=NCc2n[nH]c(=N)o2)nc2scnc12 C#CCCN=C(NCC1C2COCC12)N1CCN(Cc2ccccc2)CC1 N1(C(C2(NC(C3C4CC5C(C4)C35)=O)C(C)CCC2)=O)CC2CCC(C1)C(=O)O2 c1(CC)cccc(C(=O)NC(C2CCN(C(c3[nH]ccc3C)=O)C2)C)c1 C1(C(N2CC(OCC(=O)NCc3n(CCCC)ccn3)C2)=O)CC2(CC(=O)C2)C1 c1(CC(=O)NCC(C)NC(c2cc3cc[nH]c3cn2)=O)ccc2c(c1)CCOC2 N(C)(C(=NCc1cc(C)on1)NCC1CCN(CC)C1)Cc1cc(F)cc(Cl)c1 c1(N2CCC(CCNC(C(CC)N(C)C)=O)C2)ncnc2cc(Br)ccc12 Cc1cc(-n2cc(CCCCC#N)nn2)cnc1N c1(C(=O)NCCN(C2CC2)Cc2n(C)ncc2)cc2ccoc2c(O)n1 N1(C(CCC(=O)OC)=O)CC(=O)NC2CCCCC12 CCC(C(=O)NC1CCC(NC(c2cncc(O)c2)=O)CC1)C(C)C C1(C(N2CC3(CC(=C)C3)C2)=O)C(C2CC2)CCN1C(c1cc(C)cc(F)c1)=O Cc1cc(S(N)(=O)=O)ccc1CNC(=O)NCCc1cnnn1C c1(C(=O)NCC2C(NC(c3nnn(CC)c3C)=O)C2)cncc2ccc(F)cc12 Cc1cc(Br)cc(C(N2CC(NC(C3OCCN(C)C3=O)=O)C2)=O)c1F C1(C(=O)NCC#CCC)C(CC)CCN1C(=O)CC#N C1(CC(=O)NC2(CO)CN(C(c3c(C)scn3)=O)C2)CCC(F)(F)CC1 c1(C(=O)NC(C(C)NC(c2n(CC#C)ccc2)=O)C)cnc(O)n(C)c1=O C(CN=C(NCc1ccco1)NCC1(F)CCCCC1)=CC N1(C(CC(CN(C)C)O)=O)CCc2[nH]nc(CNC(C3(C)CC=CCO3)=O)c2C1 CC(C)CCCCC(=O)N1CC2(C1)SCCC2NC(=O)C(C)N(C)C CCC(O)C(C)C(=O)NCC1C2CC1N(C(c1cc(F)ccc1C(F)(F)F)=O)C2 C1(N=[N+]=[N-])(C(=O)NCc2c(C)cc(C)s2)CCN(C(C2CN3CCC2CC3)=O)C1 C12(NC(C3CC4CCC3O4)=O)CCCC1N(Cc1nnc(C(F)F)s1)CC2 c1(C(CNC(=O)CCCC2CC2)N(C)C(C2(F)CCC2)=O)ccc(Br)cc1 Cc1cncc(CC(=O)NCC(O)CN(C(=O)Cc2cc(C)on2)C)c1 N1(CCC(C(C)C)N)CCC(O)(C2CCC2)CC1 C1(C2CC2)(C(=O)NCc2n(C)ccn2)CCN(C(c2ccco2)=O)C1 N1(C(C(CCOC)C)=O)CC2CC(NC(=O)CCCc3cccnc3)C2C1 C12(NC(=O)CCn3cnccc3=O)CCCC1N(C(C1CSC1)=O)CC2 c1(C(=O)NCCC(C)NC(c2ccc(CC(C)C)s2)=O)ccc(F)c(CO)c1 CC(C)C(O)CC(=O)NC1CN(C(=O)C(O)C(C)C)CC1O N1(C(CC(CCC=C(C)C)C)=O)CCCCC2(C1)CN(C(=O)C=CC(C)(C)C)C2 c1(NC(C)=O)cc(C(N2CC3C(N(C)C(c4ncoc4C)=O)C3C2)=O)ccn1 C=C(C)CC(C)C(=O)NCC(C)(CO)NC(=O)CC1(O)CCOCC1 c1(NC(=O)OC(C)(C)C)cn2ncccc2n1.C12C3CCC(O3)C1COC2=O C1(C(=O)NC(C2CC=CCC2)C(=O)NCCCSCC)CCCC1O c1(OC)cc(C(=O)OCc2ncc(Cl)nc2Cl)cc2c1OCO2 N=c1cc(C(N2CCC(NC(c3ccnnc3)=O)C(F)C2)=O)c(Br)c[nH]1 C(=O)(C(C)(C)CC(F)F)N1CC(CC(=O)NC(C(C)C)CCO)OCC1 CC1CC(NC(=O)CN2CCCCCCC2=O)CCN1c1nccnc1F C1(C(N)=O)CCC(NC(C2CCCCC2c2ccccc2)=O)CC1 Cc1[nH]nc2ncc(C(N3CC(C(=O)O)C(c4ccsc4)C3)=O)cc12 C1(C(=O)NCC2C(NC(c3ncccc3Br)=O)C2)CC(C2CC2)=NO1 C1(N(C(C(C(C)C)n2cc(N)cn2)=O)C)CCC(S(C)(=O)=O)CC1 c1(OC)ccc(C(=O)NC2CCC(CNC(=O)CC3CCC4CC34)CC2)c(N)c1 N1(C(C(C)n2cccc2)=O)CCC2C1CCCN2C(c1cc(Cl)c(F)cc1Cl)=O c1(C(=O)NC2C3(CC(NC(COCC=C)=O)C3)C2)ccc(N)cc1C Cn1ccc(=O)c(C(=O)OCc2nc(-c3cnccn3)no2)c1 CCCC(C)(CCC)C(=O)N1CC2CCC2(CCNC(=O)CC2=CCCC2)C1 C1(C(=O)NCc2cncc(CC)c2)CN(C(c2cc(F)n(C)n2)=O)CC12CCC2 CC1CN(C(=O)CC2CC2(C)C)CCCN1C(C1CCC(C(N)=O)CC1)=O CCCCCC(C)(C)CNC(c1cc(Br)c(Cl)s1)c1nnnn1CCCSC c1(NC(C(C2CCOCC2)NC(C)=O)=O)cccc(CNC(=O)C(C)C2CC2)c1 C1(CNC(c2nc(C(C)=O)sc2)=O)CC(C)(C)CCC1NC(c1ccc(C)s1)=O C12(C(N(CC(N3CCCC(CC=C)C3)=O)CCC)=O)CCC(CC1)CC2 C(C(=O)NOCC(O)C(C)C)(C)(O)NC(CCCNC(C)=O)=O N1(C(C2(COC)CCCN2)=O)CC(C)OC1 N=c1ccc(C(N2C(C(=O)NCC(O)CC3CCCC3)CCC2C(C)C)=O)n[nH]1 C12(CNC(C3OCCO3)=O)CCC1CCN2C(=O)COc1cc(F)cc(Cl)c1 C(=O)(C(C)(F)C(F)(F)F)NC(C)CCNC(=O)CCc1ccc(C(C)(C)C)cc1 c1(CC(CCOC)NC(C2CCOCC2)CC)ccc(F)cc1F CC1(C)CCCCC1C(N1CCC(=CC(N2CC3(CCC3)C2)=O)CC1)=O c1(NCC(=O)NCCC(C)N(C(=O)CCC2CCOC2)C)ccccc1Cl n1(CC)nc(C(=O)N(C)CCNC(=O)C=Cc2nccs2)cc1C C1(CNC(C2CC(OC)C2)=O)CCC2(CN(C(c3ncccc3Cl)=O)C2)O1 c1(C(=O)NC2CC(C)(C)CN(C(C3CCCC3O)=O)C2)cc(F)cc2cc[nH]c12 N1(C(Cc2ccc(C)o2)=O)CCN(C(c2cc(F)ccc2N(C)C)=O)CC(O)C1 C(=O)(CCCCCS(N)(=O)=O)NCC(C)(C)OC(C(=O)OC)OCC Cc1cccc2c1OC(C(=O)NCC(C)(O)CNC(=O)CNS(C)(=O)=O)C2 c1(SCC)ccccc1C(N1CCCCC1CC(=O)NCC1CCCC(C)O1)=O Cc1nc(O)ccc1C(N1CCCC(C(=O)NC2CN(C)CC2C)C1)=O c1(C2(C(=O)NC3(COC)CCN(C(C(CC)C)=O)C3)CC2)cccc(Cl)c1F CC1CC(C(=O)NCC2CN(C(c3snc(O)c3Cl)=O)C2)Cc2nn[nH]c21 N1(C(CCN(C)CC)=O)CCC(C)(CNC(c2ccc(C)cc2N)=O)CC1 N1(C(CC(=C=C)C)=O)CC(NC(=O)C=Cc2nc(C)cs2)CC2(CC2)C1 Cc1c(Cl)ccnc1C(=O)NCCC(C)NC(C1(CC2CCCC2)CCCC1)=O C(=O)(CCC[N+](=O)[O-])NCC(C)CNC(c1ccn(C)c1)=O C1(CCNC(C(CC)N(C)C)=O)CCCCN1C(c1[nH]ncc1C#N)=O C1(N=c2[nH]c(=N)[nH]c(=NCC3C4COCC34)[nH]2)(COC)CCS(=O)(=O)C1 N1(C(c2cncc(C)n2)=O)CCC2CN(C(C3CCC34CCC4)=O)C2C1 C1(S(N)(=O)=O)(C(=O)NC2C(CNC(Cc3cnc(C)s3)=O)CCCC2)CCC1 CN1CCN(C(c2cnn[nH]2)=O)C(C(=O)NC2CC3C=CC2C3)C1 c1(C(=O)NCC2CCCN2C(=O)CCc2cccc(CO)c2)ccc([N+](=O)[O-])o1 C12(C(=O)NCC3(C(=O)NCc4ncc(CC)o4)CCCO3)CCCCC(C1)C2 N1(CC(=O)NCC2(F)CC(NC(CC3(COC)CC3)=O)C2)CCC(CO)CC1 c1(N(C)C)cncc(=NC(=O)C(=O)NCC2CCC(=O)N2)[nH]1 c1(C(C)(C)C)ncc(C(=O)NC2CCC(C(=O)CCN3CCCCC3C)C2)cn1 c1(C(N2CC(N(C(=O)C3=COCCO3)C)C2)=O)cnn2c1OCC(C)(C)C2 S(=O)(=O)(c1cnc(N2CCCC(CC#N)C2)cc1C)NCc1ccc(C)cc1F C1(C(C)NC(=O)CC2CC(C(F)F)C2)CN(C(c2nccnc2N)=O)CCO1 C(=O)(C(C)C(O)CC(C)C)NCCC1CCCN(CC(=O)NCC#C)C1 C(CC(CNC(=O)C(C)C#N)NC(c1ccc(Sc2ccccn2)s1)=O)OC C1(CC)CCN(C(=O)Cc2cnoc2)C1CNC(=O)CC1CNC(=O)O1 c1(N(CCNC(C2CC(=O)N(CC(C)C)C2)=O)CC)cncc(C#N)n1 C=C1CC2(C1)CC(C(=O)NC(CCCNC(=O)CC1CC1)c1ccccc1)C2 C(C)(C)(C(C)CC(=O)NCCN1CCOC1=O)NC(C(C)CC(F)F)=O Cc1cccc(C(C)(C)C(=O)NC(c2cn(CC3CCOC3)nn2)C)c1 c1(CC(=O)NC(CN(C)C(C2CCCC(C)(C)C2)=O)(C)C)cc(F)c(F)cc1F Cc1c(C(N2CCC2CNC(c2cn(C)nc2Cl)=O)=O)cnn1C1CCC1 N1(C(C)=O)CCCC(C2CCN(C(=O)C(C)NC3CCCC3)C2)C1 Cc1nn(C)c2c(NCc3cccc(F)c3Cl)nc(=NCC3(N(C)C)CC3)[nH]c12 N1(C(c2ccc(C)c(C)c2O)=O)CC2CCCC(C1)N2C(=O)C(C)(C)F n1(CC(=O)NCCC2CC(NC(c3c(C)noc3)=O)C2)ccc(=O)c([N+](=O)[O-])c1 Cc1cc(C(F)(F)F)c(C#N)c(=NCCN(C(=O)CCc2ncnn2C)C2CC2)[nH]1 C(=O)(CC(CC)c1ccccc1)N1CCC(N(C(C=CC)=O)CC)C1 c1(C(=O)NC(C(=O)NC(CC)COC)Cc2ccco2)ncncc1N C1(CCNC(C(C)OCCN(C)C)=O)CCN(C(=O)CCS(C)=O)CC1 c1(C(N(CC(CC)NC(=O)CCCSc2ccccc2)C)=O)cncc(F)c1Cl c1(C(=O)NCCN(C(Cc2c(CC)con2)=O)CC(C)O)cccc(OC)c1F c1(Cn2cc(CNC(C(C)(CO)OC)=O)nn2)ccc(Cl)cc1F C1(CC)(NC(c2ccc(O)c(N)n2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC1 Cc1ncc(C)c(=NCC(C)N(C)C(C2(C)CCC(=O)CC2)=O)[nH]1 C1(CCNC(Cc2nnc(C)o2)=O)CCCN(C(c2cccc(Cl)c2)=O)C1 c1(C(=O)NC2C(CNC(c3ncn(C)c3)=O)CC2)ccccc1S(=O)(=O)N(C)C c1(Cc2cc(C)[nH]n2)nc(-c2cncs2)nn1C1CCSCC1 Cc1cc(O)cc(O)c1CNC1CCC(C(N2C3CCC2CC3)=O)C1 c1(CCC(=O)NCC(CN(C)C(c2coc(O)n2)=O)O)ccc(Br)cc1 C(=O)(C(F)CCC(C)(C)C)N1C2C(NC(c3cccc(C(C)F)c3)=O)C(C2)C1 C1(CNC(COC(CC)C)=O)CC(O)C(O)CC1C(N1CC2CC1CC2O)=O C1(C(N2C(C3CCN(C(C4CN(C)C4)=O)CC3)CCC2)=O)Cc2cccnc2C1 N1(CCC(=O)NC2CC(NC(CC(C=C)C)=O)C2)C(=O)c2ccccc2C1=O C(=O)(C(F)(F)C(C)(C)O)N1CC(CC(=O)Nc2cc(CC)cc(F)c2)C2(C1)CC2 C1(NC(CCCCCCCC)=O)CCOC12CCN(C(C1(OC)CC1)=O)CC2 C1(NC(Cc2c(C)ccnc2)=O)CCCC(NC(c2cc(Cl)c(Cl)[nH]2)=O)CC1 C1(c2n(CCOC)nnn2)(ON2CCC(=Cc3cc(C)on3)CC2)CCSCC1 c1(C(=O)NC2(c3ccccc3)CCN(C(C)=O)C2)ccc2c(c1)B(O)OC2 C1(CCNC(=O)CC2CCC(=O)O2)CCCCN1C(c1cc(C2CCC2)no1)=O C=CCC(C)(C)CC(=O)N1CCCCC(NC(c2cncc3c2CCC3)=O)C1 N1(C(C(COCC)c2ccccc2)=O)CCC(c2ccc(C)cc2)CC1C c1(C2CN(C(C3CCC(n4cc(C(NS(N)(=O)=O)C)nn4)C3)=O)C2)ncccc1C c1(C(=O)OCC)c[nH]c(=NCC2CCCCN2C(=O)C(C)Cn2ccc(C)n2)s1 C(C(C)(C)CNC(=O)CC1(O)CCOC1)N(C(=O)CC1CC1)CC N1(C(C2N(C(CC)=O)CCCC2)=O)CC(NC(C)=O)C2(CCC2)C1 Cc1ccc(C(=O)NCC(N2CCCC2C(C)NC(=O)CCc2cscn2)=O)s1 N1(C(c2c(C)cnn2C)=O)CCN(C(C2COCCOC2)=O)C(C)C1C CC(C(=O)N1CCC(C(=O)NCC2(CO)CC3CC3C2)C12CC2)S(N)(=O)=O CC(C)(C(=O)N1CCC(NC(c2ccc(N)cc2Cl)=O)C1)C1=CCSCC1 c1(C(=O)NC2CC(C)N(C(C3CC=CCO3)=O)CC2)cn2cccnc2n1 c1(CNCC(C2CC=CCC2)CC)ccc(C)c(F)c1F N1(C(C2ON=C(C)C2)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 c1(CCC(=O)NCC(O)CNC(=O)C(=O)NCC2CC2)ccncn1 c1(OC)c(C(=O)NC2COCCN(C(=O)C(C)c3ccco3)C2)c(C)nn1C CCC(C)(C)C(O)C(=O)NC1COCC1NC(=O)C(C)(C)CN1CCOCC1 C(=O)(C(CCF)NC(=O)CCCn1cncn1)N(CC(=O)NC(C)C)C C1(NC(c2cccc(NC(C)=O)n2)=O)CCN(C(=O)Cn2cccc2)CC12CC2 c1(C(N2CCC(NCc3cnc(Cl)cc3Br)C2)=O)n[nH]c2cccc(F)c12 C(C(C)(CC(C)C)NC(=O)C#CC1CC1)NC(c1c(CC)nco1)=O c1(C(C)(C)NC(=O)NCC(C)NC(CF)C2CC2)ccc(F)cc1 C(=O)(C1=NOC(C)(C)C1)NCCC(C(C)C)NC(Cc1ccc(C)cc1Cl)=O CC1CN(C(C2CCOCC2)=O)CC1CNC(C1(C)CC1(Cl)Cl)=O C1(CCC(=O)NC(C)C(CO)NC(c2cnc(S)n2C)=O)CCC(=O)NC1 CC(C)CCN=C(NCc1ccc(Br)s1)NCC(c1c(Cl)cccc1Cl)O c1(C(=O)NC(C2(O)CCN(C(=O)C(F)=C3CCCC3)C2)C)ccccc1C(F)F CCCCC(CNC(C1CCCOC1)=O)NC(c1ccc(CC)nc1)=O c1(-n2c(-c3c(OC)ccc(F)c3)nc(CCCOC)n2)c(C)cc(C)cc1C Cc1cc(C)c(O)cc1C(N1CC(NC(C2CCC3(CCC3)CO2)=O)C1)=O C12(C(=O)NCCC(CNC(c3cnc(OCC)s3)=O)O)CC3CC1C2C3 C#CCC(C)C(=O)NCC1CCC1NC(C1CCCC1C(C)C)=O c1(OCC(=O)NC(CC)CNC(C2(C#N)CCCOC2)=O)c(C)cc(Cl)cc1C N#Cc1ccc(S(=O)(=O)N2CCCc3n[nH]cc3C2)cc1F C1(CNC(Cc2nc(CC)sc2)=O)CN(C(=O)C2=CCC2)CC1(F)F C(=O)(C(C)(C)C(=O)N1CC2(C1)CN(C(c1ccc(CO)c(F)c1)=O)C2)NC C12CCCC(C1)C2.C1(C(=O)NC2CCN(C(COCCC)=O)C2)C2CC3C(C2)C13 CCC(C)(C)C(O)C(=O)NC(C)CCC(=O)NCC(c1ccsc1)C c1(C(=O)NC(C(C)C)C(=O)NCc2cn(C(C)C)nn2)cc2n(n1)CCC2 C1(C(=O)NCC(N(C(C2C(SC3CCCC3)C2)=O)OC)C2CC2)CCCCCN1C N1(C(c2cnc(S(C)(=O)=O)s2)=O)CCCC12CCN(C(=O)Cc1cscn1)CC2 Cc1cccc(C(N2CCCCCC2CNC(c2cn(C)c(=O)cn2)=O)=O)c1N C(=O)(CCCC(F)(F)F)NCC12C(CN(C(c3c(OC)ncc(Cl)c3)=O)C1)C2 N1(C(c2cc(Cl)cc(Cl)n2)C(=O)NCC=C)CCOc2ccnc(Cl)c2C1 N1(C(c2ccc(OC)s2)=O)CCC(CN(C)C(c2cn(C3COC3)nn2)=O)CC1 c1(OCC)ccc(C(=O)NC(C)C(C)NC(c2cc(C3CCCC3)no2)=O)cc1 c1(C(=O)NCC(C)NC(c2ccc(OC)cc2Cl)=O)nn(C)cc1[N+](=O)[O-] C1(NC(C(c2c(C)n[nH]c2C)C)=O)CCN(C(c2ccc(C#N)cn2)=O)CC1F c1(C(N(C2CCCN(C(=O)C(C)C)CC2)CC)=O)cnc2cc(Cl)ccn12 C(CC(=O)NC1CCN(C(c2cocn2)=O)CC1O)(C(N)=O)NC(C)=O N#Cc1cccc(CNC(c2coc(CNC(C3CC(=C4CC4)C3)=O)c2)=O)n1 C(CCCCCC(=O)N1CCN2CCC1CC2)NC(C(c1ccc(C)o1)C)=O N1(C(C2C(C)N(C)CC2)=O)CC2CN(C(c3ccccc3Cl)=O)CC2(C)C1 c1(C(N2CC(C)(C)C2C(=O)OC)C(=O)NCC)nc(C)n(C)n1 C#CCC(C(=O)Nc1cnc(SC)nc1)NC(C1CC1Cl)=O CCCC(CC)C(=O)NC1CCCCC1CNC(=O)Cc1c(C)noc1Cl N1(C(Cn2c(C)ccn2)=O)CCN(C(=O)CC(C)F)C(CCO)C1 C1(NC(C2C(=C)CC2)=O)(CNC(c2cc(Br)no2)=O)CCCC1 c1(OC)cc[n+]([O-])c(C(=O)NCC(O)CNC(=O)C(c2cc(Cl)ccn2)OC)c1 c1(C(=O)NCCN(c2cnc(OCC)cn2)CCC)nc(C)c(C)s1 C1(C(N(C(C)CNC(c2cc(N(C)C)ccn2)=O)CC)=O)CCC2CC1CO2 C#Cc1cnn(C)c1C(=O)NCC12CCC(C1)N(C(=O)C(C)OC)C2 c1(CC(=O)N(CC2CCN(C(CC3C(CC)C3)=O)CC2)CC)ccc(F)c(Cl)c1 c1(C(=O)NCCOC2CC2)ccc(C(F)F)o1.C12(CCOC1)C(=O)N2 c1(OCC)c(C)cc(C(=O)NC2CC(NCc3ccccc3F)C2)cc1C C1(C(=O)NCc2cncc(OC)c2)CC(NC(=O)COC(F)F)C12CCC2 CCCC(C#N)C(=O)N1CCC(O)(CCNC(=O)CN2CCN(C)C(=O)C2)C1 CC1(C)CCCC1(O)CNC(=O)CNC(=O)CNC(=O)Cn1cc(CO)nn1 N1(C(C(C)CC2CCC2)=O)CCC(C(C)NC(C2(n3cc(Cl)cn3)CC2)=O)CC1 CC(C)CCC(C(=O)NCC(C)CC1CC1)NC(C12CCC(C1)C2(C)C)=O c1(C(=O)NCC2(OC)CN(C(C(CC)OC3CCCC3)=O)C2)cc(Cl)c(Cl)n1C C=CC(C)(CCOC)C(=O)NC(CNC(C1CC2C(C1)C2(F)F)=O)CCOC C(=O)(CCS(=O)(=O)C1CCCC1)NCC1CC(OC)CN1C(C1CCCN1C)=O c1(C(=O)NCCC(C)N(c2ncnc(C(C)(C)C)n2)C)ccc(O)nc1 C(C(C(C)C(C)C)NC(c1cn(CCO)nn1)=O)NC(CCOCC(C)C)=O C1(O)(CCNC(c2ccccc2)=O)CCN(C(C2CC3CCC3C2)=O)C1 C1(C(=O)NCC2(C)CC2)CCN(C(=O)C2C3CC(=O)CC23)O1 C(CCN=c1cc[nH]c(=NCCCC2CCCC2O)[nH]1)SCC C1(NC(c2c(C)onc2)=O)CCN(C(=O)CC2CCC2)CC1c1ccccc1 C12(CC3CCC1CC3)NC(=O)C1C(CCO1)C(=O)NC2.c1(CC)ccccc1F C(=O)(C(C)(C)C1=CCSCC1)N1CCC2(C(NC(CC(CCC)CC)=O)C2)CC1 N1(C(COC2CCN(C)CC2)=O)CC2CC1CCN2C(=O)C(O)Cc1cnc[nH]1 C1(C)(CNC(C(CC)COC)=O)COCCN(C(=O)C(C2CC2)SC)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CC2CCCC2(NC(c2ccn(C)c2C)=O)C1 N1(C(C2C(C)C2)C(=O)NCCC#N)CCC(n2[nH]c(C3CC3)nc2=S)CC1 c1(C(=O)N)cnc2ccncc2c1.N1(C(=O)NC2C(C(=O)OC)CC2)CC(F)(CF)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)C1=C(Cl)CCCC1)NC1CC(C)(C)C1 CC1(C)OCCOC1C(=O)NCCC1CC(NC(c2cc(O)ccc2F)=O)C1 C1(C(N(C2CCCN(C(C(CC)CC)=O)C2)CCO)=O)CC(=O)NC(C)C1 c1(C(=O)NCC(=O)NCCO)cc(CCNC(c2ccc[nH]2)=O)on1 c1(NC(C)=O)cccc(CCC(=O)NCCS(=O)Cc2ccccc2)c1 c1(CC(N2CCC(C(O)C)C2)=O)csc(C2CC2)n1 C(CCC(C(=O)NCCOCCOC)NC(=O)Cc1ccoc1)OC c1(C(N(CC(=O)N(C)CCNC(=O)COCCF)C)=O)cc2c(nn1)CCC2 N12CC3CC3(C1)COC2=O.C(=O)(CC=C(Cl)Cl)N(C(C)(C)C)C1CC1 Nc1ccc(Cl)cc1C(=O)NC1COCC1CNC(C1CCNC1=O)=O C1(C(=O)NCCC(C)(C)NC(c2c(CCC)n(C)nn2)=O)C2CCC(F)(F)C12 c1(NC2C(CSC)C2)[nH]c(=NCCOCCF)nc2scc(-c3ccccc3)c12 C(CCCCCCCO)=CC(=O)NC(C)C(O)C(=O)NCSc1ccccc1 C(=O)(C(CC(=O)OC(C)=O)NCCS(=O)(=O)Cc1ccccc1)OC C1(NC(C(C)n2cncn2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)O)C2 Cn1nc2cc(Br)ccc2c1-c1ccc(CN=c2cc(Br)[nH][nH]2)o1 c1(NC(=O)NC(Cc2ccoc2)CO)csc2c1CCCC2 Cc1ccc2c(ccn2CCC(=O)NC2CN(C(=O)CCSCC(C)C)C2)c1 Cc1cc(C(C)(C)NC(C2CC2NC(=O)C(C)CF)=O)cc(C)c1 C(=O)(CC(C(C)CC)NC(=O)CC1CCSCC1)NC(CCC=C)(C)C c1(CNC(c2ccccc2)(c2nnnn2C2COC2)CC)nocc1C(C)C c1(C(N2CCC(NC(CC(C)F)=O)C2)=O)ccc(COCCO)cc1 C=CC(C)(C)C(=O)NC1CCCN(C(C)C(=O)NC(c2ccc(O)cc2)C)C1 O=C(C1COc2ccccc21)NC12CCCN(C(C3CC4(C3)CC4F)=O)CC1C2 c1(C(N(CCC)CCNC(C2CCC(C)(C)CO2)=O)=O)ccnc(S(N)(=O)=O)c1 c1(CC(=O)N(CC(c2ccsc2)C)C)nnc(S)s1 CC1CCCC1(C)C(=O)NCC1CN(C(c2cnc(S)n2C2CCOCC2)=O)C1 C1(C(C)C)CN(C(=O)CSCC(=O)NCc2ccnn2C)CCN1CC(N)=O C1(CNC(Cn2c(C)cnc2)=O)CN(C(C2(CF)CCC2)=O)CCC1C n1(CC(=O)N(C(C)CCNC(=O)CC#N)C)cc2ccccc2n1 N1(C(C(C)NS(CC)(=O)=O)=O)CC2CC(CNC(C3OCCCO3)=O)C2C1 c1(C(=O)NCCCNC(CC2(COC)CC2)=O)cc(N)c(C)c([N+](=O)[O-])c1 N1(C(C)=O)CCC(CNC(c2scc3c2OCCO3)=O)C(F)(F)CC1 C(=O)(C1SCCc2sccc21)N1CC(N(C(=O)CCc2cnoc2)C)C1 C1(CNC(c2cnc3ncccn23)=O)CCN(C(=O)C(F)F)CC1(F)F C1(NC(C2(CO)CN(C(c3ccc(N)cn3)=O)C2)=O)CCOCC12CCC2.CO c1(CN2CC(NC(Cc3ccc(SC)cc3)=O)C(F)C2)cc(O)cc(O)c1 C1(C(=O)NCCN(C2CC2)CC)C(C)OCCN1C(=O)CC1CCC(C)CO1 N1(C(CC=CC=C)=O)CCN(C(=O)Cc2cc(OC)cc(C(F)(F)F)c2)C2CC12 Cc1ccc(SCC(N2CCC(NC(=O)C(n3ccc(C)n3)C)C2)=O)cc1 Clc1ccc(C2(NC3(c4cnco4)CC3)CCCCC2)cc1Cl c1(C(C(=O)NC(c2cn(Cc3ccc[nH]3)nn2)CCC)C)cccc([N+](=O)[O-])c1 CCC(CC(=O)N(C)CC1(O)CN(C(c2nc(=N)cc[nH]2)=O)C1)C(F)F CC(N=c1cc[nH]cc1S(=O)(=O)NC1(C)CCC2(CC1)CC2)c1ccncc1Cl N1(C(C(CCSC)O)=O)CC2(CCC(CNC(c3cccc4sccc34)=O)O2)C1 C(=O)(C1=CCCCCC1)NCC1C(CC)CN(C(=O)CC2C=CS(=O)(=O)C2)CC1 Cc1ccccc1C(N1CC2C(CN(C)C(c3coc(C4CCC4)n3)=O)C2C1)=O C1(C(N(CC(C)C)C)=O)CC(c2ccccc2)=NO1.n12cc(nn1)CNCCC2 C1(CC(N2CCCC(C)C2)=O)N(C(=O)COC(c2ncccn2)=O)CCC1(C)C C(CC1CCC1)(C(=O)NOCCCC1CC1)NC(c1cccc(CC)n1)=O C(C(=O)NC1C=CC(C(=O)NCc2scnc2C)C1)(C(C)C)SC C(=O)(C1CCCc2nnn(C)c21)NC1CN(C(c2c(CC)n[nH]c2)=O)CC(F)C1 C1(C(=O)OC)Cc2c(C)cccc2CN1N(Cc1cccs1)CCC(C)C c1(C(=O)NCC2(F)CC(NC(C(C#N)C3CC3)=O)C2)ccc(CCF)cc1 Cc1c(Cl)ccnc1C(=O)NCC1(CN(C(=O)C(C2CCCCC2)F)C)CC1 N1(C(c2scc(C)c2C)=O)CCN(C(C2CC2F)=O)CC12CCC2 C(=O)(C1=Cc2ccccc2C1O)NCCN(C)C(c1cccc2nc(O)oc12)=O C=CC1(CO)CCN(C(C2C=CCCN2C(c2cc(Cl)ns2)=O)=O)CC1 N1(C(C(COC(C)C)NC(C)=O)=O)CCC2(C1)CN(C(=O)CN1CCSCC1)C2 Cc1nc(C(=O)N(C(C)CNC(C2CCC(C(F)(F)F)CC2)=O)C)n(C)n1 c1(SCC)cccc(C(=O)NCC2(NC(=O)CN3CCOCC3)CCCCC2)c1 N1(C(C=C(C)C(F)F)=O)CC2C(CN(C(=O)CC(C)N(C)C)C)C2C1 C1(C(=O)NCC(C)(C(C)C)NC(C=C(CCC)C)=O)CCN(C)S1(=O)=O C(CCCCF)NC(CCOCC(C)C)=O.n12cc(nn1)CC2 N1(C(CONC(c2c(C#C)ccs2)=O)=O)CC2CC(C)C2C1 C1(NC(C2(OC)CCC2)=O)CN(C(=O)C=CC(C)C)CCC1C(F)(F)F Cc1n[nH]c(=NC(=O)N2CC3(CCN3c3nccc(C(C)C)n3)C2)n1C C1(CNC(COCC(C)C)=O)CCN(C(c2ccnnc2)=O)C12CC2 CCN(OC)C(=O)CNC(=O)NC1OC(=O)CC1(C)C CC1OC2(C(N3CC4(C3)CN(C(c3ccncn3)=O)C4)=O)CCC1C2 c1(C(N2CCCC(NC(CSCC#C)=O)C2C)=O)cn2ccn(C)c(=O)c2n1 N1(C(=O)Nc2cccc(NC(C)C)c2)C2C=CCC1CCC2.C1(C)C(=O)N1 c1(C(=O)NCCCCC(C)NC(C2CCS(=O)(=O)C2)=O)c(N)nn2ccccc12 CN=c1ccc(C(N2CCSC3CCC23)=O)c[nH]1 C1(NC(C2(C)CC3CC3C2)=O)CN(C(=O)CCC2CC(F)(F)C2)C2(CCCC2)C1 c1(OCC)cncc(C(=O)NCc2cc(C(N3CCC(C)C3C)=O)n(C)n2)c1 C1(O)(CNC(C=CC=CCCCCC)=O)CCN(C(=O)CC2CNC(=O)C2)C1 C1(NC(Cc2ccc(C)nc2)=O)CC2CN(C(C3CC4CCC3C4)=O)CC12 C1(C(C)OC)CCN(C(=O)C=CC2CCCN2C(c2n[nH]c(=N)[nH]2)=O)CC1 N1(C(C2C(C(N)=O)CC2)=O)CCC(F)(C(=O)NCCOCC(N2CCCC2)=O)CC1 C1(CC)(CNC(=O)CC2C=CC(NC(C3CCOC3)=O)C2)CC(C)(C)C1 C(=O)(CS(=O)(=O)C1CC1)NC1CC(NC(c2c(COC)nn[nH]2)=O)C1 N1(C(C2NC(=O)OCC2)=O)CCC(C(=O)O)C(N)C1 C1(CC(=O)N(CCC(=O)OCC)C)CCN(C(c2nonc2CC)=O)CC1 C=C1CC(C(F)(F)F)(C(N2CC(O)(CNC(C3CCCCS3)=O)C2)=O)C1 C12(O)CC3(CCCN(C3)C1=O)C2.c1(C(=O)OC)onc(C)c1OC c1(CNC(C2(CCC=C)CN(C(=O)C(c3ccsn3)C)C2)=O)cccc(C)c1 c1(C(N(CC(=O)NC(c2nccs2)CC)C2CC2)=O)cnccc1N(C)CC Cc1ccc(C)c(NC(=O)CC2CCC(CNc3ncc(C)c(C)n3)CC2)n1 N1(C(C=CC)=O)CCC(c2ccccc2)(NC(=O)C(CC)OCC)C1 C1(CC#C)CCN(C(=O)C(CCC)NC(=O)Cc2cc(C)cs2)CC1 c1(C(N(C(CCNC(COC(CC)C)=O)C)C)=O)c(F)ccnc1Cl Cc1nn(C)c(C)c1C(=O)NC1CCCCC1C(N1CCCC(CO)C1)=O C(=O)(C(F)CCC(C)C)N(C)CC1CCN(C(C2CC(CC)OCC2)=O)CC1 O=C1CC(C(=O)N2CC3(C2)CN(C(C2CC4CCC4C2)=O)C3)c2ccccc21 Cc1nc(N2CCC(NC(c3sccc3C(F)F)=O)C2)ccc1C#N Cc1ccc2c(CCC(N3CC(F)(CNC(C4CC4(C)C(C)C)=O)C3)=O)c[nH]c2c1 CC(O)CN=c1[nH]c(=NCCCC2CCCCO2)c2[nH]ccc2[nH]1 CC#CCC(C(=O)NCC1CC2CCCC2C1)NC(=O)C(CO)N(C)C C1(C(C)(C)C)CC(CNC(C2(F)CCCC2)=O)CN(C(=O)C2CC2)C1 C(=O)(CCC1=CCCCC1)N1C(C)(CC(=O)NCC2(C)N=C(C)SC2)CC1 C1(NC(C(CO)OC)=O)COC2CN(C(=O)CC3CCSC3)CC12 C1(CNC(C2(SCC)CC2)=O)CCCCCN1C(=O)CCc1cn(C)cn1 N1(CC(COCC(C)C)O)CCC(C)(NC(c2cnc(Cl)c(Cl)c2)=O)CC1 C1(C(=O)NCCC2(CNC(C(=O)NC(C)C)=O)CC2)CS(=O)(=O)CC12CC2 CC(N=c1[nH]c2cc(Cl)ccc2s1)C1CCCCN1C(=O)C(F)C1CCC1 Cc1ccc(CC(N2CC(NC(c3c[nH]nc3C3CC3)=O)C3(CC3)C2)=O)c(C)c1 CC1=C(C(=O)NCC2CC3(CC(NC(=O)C(C)Sc4ccccn4)C3)C2)CCC1 CCC(C)(COC)C(=O)NC(C1(O)CN(C(=O)CSCC(C)C)C1)C CC1CCCN1C(C1C(NC(=O)C(C2CCCCC2)=O)C1(C)C)=O Cc1ccc(C)c(C(N2CCC(N(C(=O)CC3(CC(=O)NC)CC3)C)C2)=O)c1C N1(C(CC=CC)=O)CCN(C(c2ccnc(C3CCC3)c2)=O)C(C(F)F)C1 C1(O)(CNC(CSCCC)=O)CC(C)(C)C1.C12(C)CC(C1)NC2=O c1(C(C)NC(c2c(C)n(CCO)nc2)=O)ccc2c(c1)CC(=O)N2C c1(CC)ncc(C(N2CC(NC(C3CC34CCOCC4)=O)CC(C)C2)=O)c(O)n1 c1(C(=O)OC)cc(O)c(Br)cn1.C12CCCCN1S(=O)(=O)C2 CC1CN(C(=O)C(F)CC2CCOC2)CC1NC(C1CCNC(=O)C1)=O Cc1nc(C=CC(N2CCCC2CNC(=O)C(C2CC(F)(F)C2)N(C)C)=O)cs1 C(=O)(CC(C)n1ccc(C)n1)NC(C1CC(NC(COCCCCC)=O)C1)C c1(C(=O)NCC2OCCCN(C(C3C(C)CCO3)=O)C2)cccn2[nH]c(=N)nc12 c1(NC(=O)NC2C(c3ccc(Br)cc3)(C)C2)cc2cccc(Br)c2nc1Cl C1(C(C)(F)F)(C(=O)NC2(C)CN(C(C(C)NC(N)=O)=O)C2)CCOCC1 C=C(C)CCCC(=O)NC1CCCC1CNC(=O)C(C)CCOC Cc1cnc(NC(c2cccc(Cl)c2)C)c(S(=O)(=O)N2CCC(CO)CC2)c1 c1(C(=O)NCCCCN(C(C2(C(=O)OC)C=CCC2)=O)C)cccc2ncsc12 C(=O)(C(F)(F)CC(C)C)N(C1CCCN(C(c2cccc(OCC)c2)=O)C1)C N1(C(C2C(C)=CCC=C2)=O)CCC2(CC1)CCN(C(=O)CCc1ccoc1)CC2 N1(C(Cc2c(C)snc2)=O)CCc2cc(-c3cn(C4CC4)nn3)ccc21 c1(NC(c2cnn3ccc(C)cc32)=O)n[nH]c(=NC(CO)C(C)CN(C)C)s1 C(CCC(C(=O)NNc1cccnc1)NC(=O)OC(C)(C)C)OC C1(NC(C(C)OC)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC1F C1(NC(C2CCN(CC#C)CC2)=O)COCCN(C(C2CC3CCC2O3)=O)C1 c1(OC)ccc(C(=O)NCC2C=CC(NC(C3CCCS3(=O)=O)=O)C2)nc1Cl c1(CC)noc(C(=O)NC2CCCC2CNC(=O)C(c2ccc(Cl)s2)=O)n1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(NS(NC)(=O)=O)CC1.C1(=O)CO1 Nc1ccc(C(=O)NC2CN(C(c3cnc(O)o3)=O)CCC2CO)cc1O N1(C(Cc2cccc(CC)c2)=O)CC2CC(C1)N2C(c1ncncc1C)=O c1(C(N2C(C(C)NC(=O)CC3CCC34CCC4)CCC2)=O)cnn2ncccc12 CC1C(=O)OCC1C(N1CCCC(c2n[nH]cc2C(=O)OC(C)(C)C)C1)=O N1(CC)CCC(NC(c2ncoc2CNC(=O)C(C)(O)C2CCC2)=O)C1 N1(C(CCSCC)=O)CC(F)(F)CC1(C)CNC(c1ccc(NC(C)=O)cc1)=O CCC(C)C(O)C(=O)NC1CCC(NC(c2ccco2)=O)C1 CCC(C)(C)CC(=O)NCC(C)(F)CNC(=O)C=Cc1ccsc1 CCC(C)C(C(=O)NC1CC(CCC(=O)NC2CCC(C(C)O)CC2)C1)N(C)C c1(N(C(C(=O)NC(CC#C)CC#C)=O)C2CCC2)ccccc1C#C C1(CF)CN(Cc2cn(C3CCCC3O)nn2)CCO1 C(C)(C(C)(C)C(=O)N1CCCC(OC)C1C)NC(c1n(CC)nnc1)=O c1(Nc2scc(C(N(CC(=O)NCC(N)=O)CC)=O)n2)cc(Br)ccc1SC N1(C(CCOC(C)=O)=O)CCC(NC(c2cc3c([nH]2)CCCC3)=O)C12CCCC2 C1N(C(C2(c3nn[nH]n3)CCCOC2)=O)CCCC12CCC2 Cn1nc(CCC2CCC(NC(=O)NC3CC3Cl)CC2)cc1-c1cccc(F)c1 c1(C(=O)NC2CCC(N(C(=O)CCc3ccsc3)C)C2)ccc(Cl)c(F)c1O c1(C(N2CCC(CNC(c3ccc(O)cc3)=O)C2)=O)ccc[n+]([O-])c1 C1(NC(CN(C)CC)=O)CN(C(c2ccc(-c3cnc[nH]3)cc2)=O)CC1C C(CO)(C(=O)NCC1CCC1C(=O)NC1CC1CN(C)C)OC C=CC(C)(C)CC(=O)N1CCC(NC(C2CC23CCSCC3)=O)CC1C N#Cc1ccc(C(=O)NC2CCCCC2NC(C2CCOCC2)=O)nc1 C(=O)(CC(C)C(=O)OC)N(C)CC1CCN(C(Cc2cccc(C)c2)=O)C1 c1(C(N2CCC(CNC(C(C)NC(=O)C3CC3)=O)C2)=O)cccc(C(C)C)c1N Cc1nc2cccc(C(=O)N(CC(C)NC(=O)C=Cc3cncnc3O)C)c2[nH]1 n1(CCC)cc(C(=O)NCCCCNC(C23CSCC2C3)=O)cn1 C1(C(N2CC(=C(CNC(c3cc(C(F)(F)F)no3)=O)F)C2)=O)C(F)(F)C12CC2 C1(OC)CCCN(C(=O)CC2CN(C(=O)C(C)NC(N)=O)CC2C)C1 Cc1c(C=CC(=O)NC2(CCCNC(C3COC(C)C3)=O)CC2)cnn1C C1(CNC(C2(C)C(C)OCC2)=O)CCN(C(=O)CNC(=O)C(C)(C)C)C1(C)C c1(C(N(CCCN(C)C(C2CC2CF)=O)C)=O)cc2c(nc1O)CCC(C)(C)C2 CCC(C)CCC(=O)NC(Cn1cccn1)C(=O)NCC1(C)CCOCC1 N1(CCC)C(=O)CCC1C(=O)N(CC(N1CCN(C(C2CC(C)C2)=O)CC1)=O)C C#CC1CCCN(C(C2CCC=CC2NC(C2CC(=O)C2(C)C)=O)=O)CC1 C(CCF)(C(=O)NCCCNC(=O)OC)NC(C(CC)=CCCC)=O N1(C(CCc2cccc(OC)c2)=O)CC2(C1)CN(S(=O)(=O)c1cccs1)C2 C1(C2CC2)(CNC(C(C=C)C)=O)CCN(C(c2cc(CC)nnc2C)=O)C1 C(=O)(C(C(C)C)C(C)C)NCCCCCN(C(CNC(=O)OC)=O)C CC(C(=O)N1CCN(C(c2cnc(N(C)C)nc2)=O)C(CC(F)F)C1)P(C)(C)=O C1(NC(CC(C=C)C)=O)CN(C(=O)CC2CCC=CCC2)C2CCCCC12 C1(C(=O)NCCC2(O)CN(C(=O)C3=CCCCC3)C2)CC2CCCC2C1 N1(C(c2cnc(OC)nc2C)=O)CC(NC(=O)CCCCCF)C(C2CC2)C1 c1(CC)cc(C(N2CCCOC(CNC(C3CC4CCC3C4)=O)C2)=O)cc(O)n1 c1(C(=O)NCCNC(c2sc(Br)cc2F)=O)cc2c(cn1)COCC2 C1(NC(CCc2nc(C)sc2)=O)CCCN(C(=O)CC2C=CS(=O)(=O)C2)CC1 C1(C(N2C(CN(C(CNC(CC)=O)=O)C)CCC2)=O)CCCN1N=O C(CN=C(NCC)NCC(C)(C)N(CC1CC1)CC)(c1ccccc1)OCC C1(C(N2CCC3(CC2)CC3)=O)CCN(C(=O)c2ccncc2F)O1 C1(C(N2CCC(N(C)CC)C2)=O)CC(NC(C2CCCC2O)=O)C(O)C1 c1(OCC)cccc(CN2CCCC2CC(N2CCC3(CC2)CC3)=O)c1OC c1(C(N2CCC(N(C(Cc3cn(CC)nc3)=O)C)C2)=O)sc2ccsc2c1C CC(C)(CN=c1[nH]ncs1)NC(=O)CSc1ccccc1Cl N1(C(C2(C)CC(F)C2)=O)CCCCC(C(N2CCC(OCC(N)=O)C2)=O)C1 N1(C(CCC#CC)=O)CCC(C)(C(=O)NCC(C)COCC)CC1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(CNC(C(COC)(C)C)=O)OCC1 C1(OC(C)C)CCC(c2ccccc2)CC1.C12CCCN1C2=O C1(C(C)C)CCC(n2nc(-c3cnn(C)c3)nc2-c2ncn(C)n2)CC1 C1(CC(=O)N(CCC=C=C)CC)CC(O)C(O)CC1NC(=O)CSCCC(C)C c1(OC)ccnc(CN(CC(=O)NC23CC(F)(C2)C3)C)c1 c1(C(=O)Nc2ccc(-n3ccnn3)cc2)ccc2c(c1)CNCCN2 C1(c2c(CC)cccn2)CCCCC1C(=O)OC(C)(C)C.C12CCN(CC1)C(=O)N2 C(=O)(CCC(F)(F)C(F)F)N1CCCC(O)(CNC(CC(=C=C)C)=O)CC1 C(CC(C)C(=O)NC(CNC(C1(c2ccn(C)n2)CC1)=O)CC)=CC N1(C(C(C)C#N)=O)CC(O)(C2CCN(C(=O)COc3c(F)cccc3F)CC2)C1 c1(C(N(CCCN(CCC(=O)OC)C(C)C)C(C)CO)=O)ncccc1O C1(C(N2CCN(CCn3cc(SCC(C)O)nn3)CC2)=O)CC2COCC(C1)C2 CC1CCN(C(C2(CCF)CCOCC2)=O)C1CNC(=O)Cc1ccsc1Cl c1(COC)ccc(S(=O)(=O)N2CCC3(CC2)CC3C(=O)O)c([N+](=O)[O-])c1 C=CC(C)CC(=O)NC1(C)CN(C(=O)CCOc2ccc(CC(N)=O)cc2)C1 N1(C(CCOCC)=O)CC2(CC1CNC(=O)CCCCOC)CC2(F)F CC(C(=O)NC1CC(O)CN(C(c2ccncc2Br)=O)C1)S(N)(=O)=O c1(C(=O)Cc2ccccc2F)ccc(Cl)cc1Cn1cc(CC(O)C2CC2)nn1 Cc1cccc(CC(N2CCCC(C3CC3)(NC(=O)CN(C)C(N)=O)C2)=O)c1Cl C1(C(=O)OCC)CCN(C(=O)C(Cc2ccc(C)cc2)NC(C)=O)C1C N#Cc1cnn2cc(C(=O)NC3CCCN(C(c4ccccn4)=O)C3)cnc12 C1(C)(CNC(C(CC)SC)=O)CCC(NC(c2cc(C(C)C)[nH]n2)=O)CC1 c1(C(=O)NC2CN(C(C34OC(C)(C)C(C3)C4)=O)C2)cnn2ncccc12 N1(C(C(CC)C)=O)CCOC2(C1)CN(S(=O)(=O)c1sccc1OC(F)(F)F)C2 CC(C)CC(CNC(c1ccn(CCNC(C2(C3CCCO3)CC2)=O)c1)=O)CO C1(NC(CC(C=C)CC)=O)CN(C(=O)CCC2CCCC2)CCC12CCOCC2 CC(O)(CC(=O)NC1(CNC(c2cccc(N)c2)=O)CCCC1)C1CC1 c1(NC(=O)OC)ccnc2ccc(C(N3CCCCC3C(O)C(F)(F)F)=O)cc12 c1(C(=O)NCc2ccc(CC)c(F)c2)c(O)cc(=O)n2c1CCNCC2 C=CCC(CNC(c1ccoc1CNC(C1(C)CC=CCC1)=O)=O)CC(C)C CC(C)C(F)(CNC(C1(NCCN(C)C)CC1)=O)C(=O)N1CCCCCC1 C1(CN(C(COCC)=O)C)C2CN(C(=O)C(c3ccc(F)cc3)(C)F)CC12 c1(C(C(=O)NC2CC(NC(c3ccc(OC)nn3)=O)C2)O)cc(F)c(F)c(F)c1 CC1(C)CN(C(c2nncs2)=O)CC(CNC(=O)CC2CCOC(C)(C)C2)O1 c1(OCCC(=O)N(C)CC2CCCN(C(C(CC#C)C)=O)C2)ccc(F)cc1Cl C(=O)(C1OCCc2ccccc21)N1CCCCCC(NC(c2ccco2)=O)C1 C12(O)CCCN(C1)C2=O.C1(OC(C)(C)C)CC(F)(F)C1.C1(CC)CCCC1C(=O)O C1(NC(CCC(=O)NC)=O)CCC(C)N(C(c2ccc(NC=O)cc2)=O)C1 C=CCCCCCCC(=O)NCc1ccnc(C(=O)N(CCCCO)C2CC2)c1 CC1(C)CC(C(=O)NOCC2CCOC2)CN(C(=O)CCCC(F)(F)F)C1 C(CCCCC(=O)NC1CN(C(=O)Cc2cccc(F)c2)C2CC12)N(C)C CCC(C)CCC(=O)NC(C1(C(=O)NCCCn2ccnn2)CC1)C N1(C(CC(=O)NCC#C)=O)CCC(C2CCCN2C(=O)C(F)C2CCC2)CC1 N1(C(CC=C)=O)CCC2(CCCC2C(N2CCC(C)(C)C2)=O)C1 C1(NC(COCCC)=O)CCOCC1C(=O)NC(c1ccn(C)n1)CC C1(Cc2cn(CC(=O)NCCCS(C)=O)nn2)CCC(C)(C)CC1 c1(C(=O)NCC(=CC(N2CC(C(CC)C)C2)=O)C)cnncc1O N1(C(CC)=O)CCCC1C(=O)NC1CC(N(C(=O)C(C)C2CCOC2)C)C1 N1(CCC)C(=S)NC(c2cc(O)cc(Br)c2)C2=C1CC(C(=O)O)NC2=O C(=O)(C(C(C)NC(C1CC2C=CC1O2)=O)C(C)C)NCCc1c(C)ocn1 C1(NC(CCCCC(CC)C)=O)CCOC12CCN(C(=O)CC(C)C)CC2 C(=O)(CS(=O)(=O)C1CCCC1)NCCC1CC(NC(c2ccc(C#C)o2)=O)C1 C1(C)(CNC(c2cc(OC)ncc2)=O)CCCN(C(C2CC(=O)C2(C)C)=O)C1 N1(C(C2N(C(c3ccnc(C)c3N)=O)C(C)C2)=O)CCOC2COCC2C1 N1(C(c2ccc(C)n2C)=O)CCC(NC(C2CCOC2)=O)C(F)(F)CC1 N1(C(C(C)(C2CC2)OC)=O)CC2CCCC(CNc3nccc(C)n3)C2C1 N1(C(C2(C#N)CCCC2)=O)CCCC(CO)(NC(C2CCCCO2)=O)C1 C(=O)(CCCCCN(C(=O)CC(C)(C)C)C)N(C)CC1CC1c1ccco1 CC(C)CC(C(=O)N1CC(c2c(Cn3cc(C4CC4)nn3)nn(C)c2)C1)N(C)C C(CC(C(=O)Nc1ccccc1CC(C)C)NC(=O)OC(C)(C)C)SC N1(C(C2C(C(C)(C)O)C2)=O)CC(O)(CCNC(c2csc(-c3cnc[nH]3)n2)=O)C1 Cc1c(C(=O)NC(C2CCCN2C(=O)CCSCC(N)=O)C)ccn1CCO C=Cn1nccc1C(N1CCC(CN(C(=O)C(C)SC)C)C1)=O N1(C(c2n(CCC)ncc2)=O)C2CCC1CN(C(C1CCOCC1)=O)CC2 C(=O)(C(CNC(=O)C(C)CC=CC)(CC)CC)NC(C#CC)(C)C N1(C(c2ncn(CC)n2)=O)C2CCC1C(F)C(NC(c1coc(C(C)C)n1)=O)C2 Cc1cc(=NC(=O)C(=O)NCC(c2cc(F)cc(Cl)c2)NC(=O)C=CC2CC2)[nH]o1 C(C(C)(C(=O)N1CC2C(N(C)C(c3cc(Br)n(C)c3)=O)C2C1)OC)OC c1(C(N(CCCNC(C2C3CCC(=O)C23)=O)CC)=O)cccc2c1CCCC2=O Cc1cccc2c1OCC2C(=O)NCC1(C)CCN(C(c2cc(C)n(C)n2)=O)C1 c1(CN2CCN(C(c3cc(F)ccc3Br)=O)C(CO)C2)c[nH]c2c(F)cccc12 N1(C(CC2(OC)CCC2)=O)CCC(NC(=O)C(C)Cc2ccccc2)C(O)C1 C1(C(N2CCC(N(C(CC)=O)C)C2)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1 c1(C(=O)OCC)sccc1C(=O)N(C1(C(=O)NC2CC2NCC)CCC1)C C1(C)(CC(=O)NC(C(C)C)CNC(C2CCOC2)=O)CC(F)(F)C1 Cc1cc(NC(=O)CCc2nc(C(F)(F)F)n[nH]2)nc(N(CC(C)C)C)n1 C(CCC(=O)NC1CCCC1NC(C1CCN(CC(C)C)C1)=O)=CCC=C c1(C(N(CC(C)NC(=O)CCc2ncccn2)CC)=O)cccc([N+](=O)[O-])c1Cl C1(CNC(=O)C(F)n2ccnc2)C2CC1N(C(c1cccc(C(F)(F)F)c1)=O)C2 c1(N2CCC(N(C(=O)CN3OC(C)(C)CC3=O)C)C2)c(C)cncc1[N+](=O)[O-].CN c1(C(=O)NCC(C)CNC(c2cncs2)=O)ccc(CC(C)(C)C)cc1 c1(C(C)NCC(c2cccnc2)OC)ccc(Br)c(Cl)c1 c1(CN(C)C(c2conc2CNC(=O)CCC2(C)CC2)=O)ncccn1 c1(N2CCOCC(C(=O)NC(CCCC)C)C2)nc2ccccc2s1 Cc1cc(C(=O)NCCC2CCN(C(=O)C=CCO)C2)n2nc(C)c(C)c2n1 c1(C(=O)NCC(CC)NC(c2cc(C)ncc2C)=O)ccn2c1CSCC2 N1(C(CCCCC=C)=O)CCC2(NC(=O)CCS(C)=O)CCCC12 C1(C)(C(=O)NCc2c(CCNC(c3ccc(CC)s3)=O)ocn2)CCCOC1 N1(C(c2cc(Cl)cc(C)c2N)=O)CCN(C(c2nccnc2N)=O)CC(C)(C)C1 C12CCC(CC1)N(CC)C2=O.c1(C(CC)OC)cn(Cc2cnns2)nn1 c1(C(=O)NC(C(C)NC(CNC(CC)=O)=O)C)cnc(C)cc1C NC1CN(CC(C2CS(=O)(=O)C2)=O)CC(F)(F)C1 CCCCCCCCCC(=O)NC1C2CCN(C(=O)C(=O)C(C)(C)C)C12 C1(NC(c2cnc(Cl)s2)=O)CC2CC1N(C(c1ccc(-c3ccco3)s1)=O)C2 C1(CC)CCC(C(=O)NCC(CNC(=O)C(C)(C)c2cnsc2)OC)CC1 C1(C(C)C)CN(C(C2(C)CCCN(C(C3CN(C(N)=O)C3)=O)C2)=O)CCCO1 c1(SC)nc(Cl)cc(=NC2CCN(CC(=O)NCC3CC3)CC2)[nH]1 O=C(C1=NOC2(CCN(S(=O)(=O)C3CC3)C2)C1)Nc1cc(F)ccc1N1CCCC1 N#Cc1cc(I)ccc1NNC(=O)N1CCC(C(O)C(N)=O)CC1 Cc1[nH]c(=N)nc(O)c1CC(=O)NCC(C)CNC(=O)CC1CCC(F)(F)CC1 C1(CN(C(C2C(CC)C2)=O)CC)CCN(C(=O)C(c2ccccc2)N(C)C)CC1 c1(CNC(CNC(c2cccc(CCOC)c2)=O)=O)ccc(C)cc1OC c1(C(=O)NC2C(C=C)CN(C(C3(C)CCCO3)=O)C2)nccn2cc(C)nc12 C1(C(=O)NC(CCC)C2CCCC2)CCN(C(=O)CC(C)CCC)C(C)(C)C1 CCCC(CC)C(=O)N1CCOC(CCNC(c2coc3c2CSC3)=O)C1 C#CCC(C)(C(=O)NC(c1ccc(O)nc1)C)NC(=O)C(C(C)C)NC=O c12ncnc(c1N)NN2C.C1(N)CN(C(=O)OC(C)(C)C)CCC1C.C(C)(C)(C)O c1(C(N2C(C)(C(N3CC4C(C3)C4(C)C)=O)C=CC2)=O)cccc(F)c1F c1(C(=O)NC2CCN(C(c3cccc(F)c3O)=O)C23CC3)cncc2ccsc12 c1(C(=O)NCCC2(OC)CN(C(c3cnn(C)c3)=O)C2)cc(C)nn1C c1(CNC(c2c(C)scn2)c2nnnn2-c2ccccc2)cccc(C(N)=O)c1 C1(NC(Cc2c(C)cc(C)s2)=O)CC(NC(=O)CC(C)(C)C2CC2)C(O)C1 N1(C(c2c(C)cc[nH]2)=O)CCOC(CCNC(C2CCCN2C=O)=O)C1 c1(C(=O)Nc2scc(-c3c(C)cc(O)cc3)n2)cc(F)c(F)c(Br)c1F C(C)(CCC(=O)N1CCOC(C(=O)NCO)C1)N(C(C)=O)C.c1(C2(N)CC2)ccccn1 c1(-c2cn(CC3N(C(C(C4CCOCC4)OC)=O)CC3)nn2)cncc(C)n1 c1(C(=O)NCC(CN(C(c2n[nH]c(C)c2Cl)=O)C)C)ccc2c(n1)CCC2 c1(NCC(CC)Oc2cccc(Cl)c2)cc(NC2CCCCC2C)ncn1 N12CCCC(C1)C(=O)NC1CC(C1)NC2=O.C(=O)(C(O)c1ccsc1)NC1CC1 c1(CNC(C2(C(C)C)COC2)=O)ccc(C(=O)N(C2CCOCC2)C)[nH]1 N1(C(c2c(OC)scc2)=O)C2CCC(C(=O)NCC(C)(C)C(O)C(C)C)C1CC2 C1(C(=O)NCc2scc(C(=O)NCc3occ(C)c3)c2)COCC(C)O1 N1(C(C(c2cccs2)OC)=O)CCCN(C(c2cc(-c3ccco3)co2)=O)CC1 C(=O)(C(CC(C)C)N(C)C(C1OCCCO1)=O)N(C)Cc1ccc(C)cc1 CC1(CNC(=O)CC2CC2)CN(C(c2nccnc2-c2ccncc2)=O)CCO1 Cc1cc(=NC(CCO)C2CCCCO2)[nH]c(C)c1C#N CCC(C)C(=O)NC(c1ccccc1)C(=O)NCC1(C)CCOC1 c1(N(C)CC2(CC)CCCC2)nc2c(c(=NC3CCC(C)CC3)[nH]1)CCCCC2 C#CCCCCC(=O)NCC1C2CN(C(=O)CCSc3c(C)noc3C)CC12 C=C(C)C1CN(C(C2CC3(CCN(C(C4CN(C)C(=O)N4)=O)C3)C2)=O)CCO1 C1(C)(C(=O)NC2(COC)CSC2)CN(C(=O)CC2(C)CCOC2)C1 N1(C(=O)CC2OCCO2)CC2(CC2C(N2CCC(c3cc[nH]n3)C2)=O)C1 Cc1ccc(C)c(NC(C2(NC(c3cc(C)c(C)[nH]3)=O)CC(O)C2)=O)c1 C(=O)(NNc1ccc(C#N)c(F)c1)N1CCC2(CCC(c3ccc(OC)cc3)C2)C1 C1(C(C)C)CCN(C(=O)C(C)NC(=O)CCCC2CCCO2)C1 N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CCNC(C1CC(C)CCO1)=O C12(NC(=O)COCC3CC3)CCC(CC1)N2C(=O)C(=O)Nc1ccc(Cl)cc1 C1(C)(CC(=O)NC(C(C)(C)C)CNC(=O)Cc2cc[nH]n2)CCS(=O)(=O)N1 C=C(C)CCC(=O)NC1CCCN(C(=O)C(O)CN2CCOCC2)C1 C1(C(=O)NC2CC(CCNC(CCOCC(C)C)=O)C2)CCc2nncn2C1 N1(C(C(C=CCCC)O)=O)CCCN(C(=O)Cc2c(C)noc2Cl)CC1C Cc1cn(CC(N2CCC2(C)C(N2CCOC3CC23)=O)=O)c(=O)nc1O Cc1nc(C(=O)NC2C3CN(C(c4cc(C)c(Br)s4)=O)CC23)c(C)o1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC(CNC(C(CC)CC)=O)C(O)C1 CN1C(=O)Cc2cc(S(=O)(=O)NCC3CCCC3C(=O)O)ccc21 CCC(C)CC(=O)NCc1cc(C(=O)NC(C)Cc2cn[nH]c2)co1 c1(C(N2CC(C(F)(F)F)CC(C(=O)OC)C2)=O)cccc2c1CNC2=O c1(N2CCCC(C(=O)NCC(C)NC(CC)=O)C2)nc(C)ccc1CC C1(C(N(C(CC(=O)OC)C)C)=O)CCN(C(C23CCC(C2)C3)=O)C12CC2 c1(C(=O)NCCC2(CNC(COCP(C)(C)=O)=O)CC2)cncc2[nH]ccc12 N1(C(CC(C)C)=O)CC2CCCC2(CNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(=O)NC(C2CN(C(C3CCC(=O)O3)=O)CC2O)C)[nH]nc2c1COC2(C)C C1(C(N(CCc2ccc(C)cc2)C)=O)C2CC(CC2F)N1C(C1CC1C1CC1)=O C1(C(=O)NC2CC(C)(NC(CCc3cn(C)nc3)=O)C2)CCC(C)(C)OC1 N1(C(c2c(CC)ncs2)=O)CC2N(C(=O)Cc3ccoc3)CCC2(C)C1 Cc1cccc(C(N2CCC(NC(=O)CC3CCCC3(F)F)C(O)C2)=O)c1Cl c1(-n2cc(CC(C3CCCN(C(C4CC5CC5C4)=O)C3)=O)nn2)ccc(F)cc1 C(CC)(CC)(CCNC(c1scnc1C1CCCC1)=O)NC(CC(C=C)C)=O N1(C(C(=O)NCC(CC(=O)NC)C)=O)CCC2(COCC(CO)O2)C1 Cc1cc2c(C(N3CCCN(C(c4oc(C)cc4C)=O)CC3C)=O)nccn2n1 c1(C(N(C2CCN(C(c3csc(CO)n3)=O)C2)CC#C)=O)coc(C(=O)OC)n1 N1(C(=O)C2COc3ccccc32)Cc2ccccc2Sc2ccccc21 N1(C(CCSCCCC)=O)C2CCCC1CC(NC(=O)CC1CCC3CC3C1)C2 S(=O)(=O)(c1ccc(C(F)F)c(F)c1)Oc1cc(C)c(CNCCC(C)C)cc1 c1(CC(=O)NC2C3CN(C(C4(C#N)CCCC4)=O)C(C3)C2)ccc2c[nH]nc2c1 C(=O)(CCCC(=O)OC(C)(C)C)NCC1CC(NC(CC(C)N(C)C)=O)C1 c1(C(C2CCCC2)NC(C(C2(C)CC2)NC(CNC(=O)OC)=O)=O)ccccn1 C1(O)(CC(=O)N(CC(CN(C(=O)CSCc2ccccn2)C)O)C)CCOC1 c1(OC)cc(Br)cc(CN2CC(OC)CC(NC(=O)OC(C)(C)C)C2)c1OC c1(OC(C(=O)NCC(=Cc2ccccc2)O)(F)F)ccccc1F.c1ccccc1 c1(C(N(C2CCN(C(C3CC3F)=O)CC2)CC(C)C)=O)nnn2c1CSCC2 c1(SCC(=O)N(C)Cc2cccc(C)c2)cc(Cl)cc(Cl)c1Cl C1(CO)CC12CC(NC(c1nnnn1C(C)C)(C)CC1CCCC1)C2 N1(C(Cc2c(C)nc[nH]2)=O)CCCN(C(=O)C=C(Cl)Cl)C(C)C1.C(C(C)(C)O)NC CC(F)(C(=O)Nc1cccc(NC(c2ccc(S(N)(=O)=O)o2)=O)c1)C(F)(F)F c1(OC)ccc(Cl)cc1CN1CCCOC(CNC(c2ccc(Cl)nc2O)=O)C1 C1(NC(C2CCC2)=O)CCCC12CN(c1cc(Cl)nc(C(F)(F)F)n1)C2 c1(C(N2C(CCNC(=O)CC3CSCCS3)CCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1cc([N+](=O)[O-])cnc1NCCC1CC(NC(c2cncn(C)c2=O)=O)C1 C1(NC(C2CC(C(C)C)C2)=O)CCCC(Nc2nc(-c3ccccc3)ns2)C1 c1(SCCOCCOCCNC(CCOC2(C)CC2)=O)ccccc1CC#N CCCC(CC)C(=O)NCC(C)(CC(C)C)NC(c1ccc(C2CC2)c(F)c1)=O c1(C(=O)NC)ccnc(-c2ccc(C(=O)Oc3sccc3OC)cc2)n1 c1(C(C(=O)NCC(CN(C(C=CC)=O)C)O)C)ccc(C(F)F)cc1 c1(C(=O)NCCCN(C(=O)CNC(=O)Nc2ccccc2)CC)ncncc1Cl c1(OCC)cc(NC(=O)NCCc2c(Cl)cccc2Cl)ccc1Br N1(C(c2cnc(C(C)C)s2)=O)CCOCC1CCNC(=O)C(C1CCOCC1)F C1(CC(=O)NC(C)CCNC(=O)CCc2cncc(O)c2)CCC2(CCC2)O1 C(c1c(F)cccc1F)=CC(=O)NCC(CN(C)C(C1CC1C(C)(F)F)=O)O N1(C(CN2CCC(C)C2)=O)C2CC=C(C(=O)N3CCC3CC3CCCC3)C1CC2 CC1CON(C(=O)c2cccc(C3SCCS3)c2)C1 C1(C(C)C)(C(=O)NC(CNC(=O)C(C)(C)OC(C)(C)C)C2CC2)CCCO1 Cc1ccc(C(C)(C)C(=O)NCC2(NC(C3CCC4CCC34)=O)CC2)cc1 C12(C(N3CCC(N(C(C4CCC(C)(C)O4)=O)CC)C3)=O)CCC(N=[N+]=[N-])(CC1)C2 Cn1c(C(=O)NC2(C)CN(C(C3CCCC(O)C3)=O)C2)cc2sccc12 c1(C(=O)NCC(CO)NC(C(=O)NCCOC)=O)cnc(O)n1C N1(C(C=CC=CC)=O)CC2(CNC(c3occc3Br)=O)CCC1C2 CC(N=c1[nH]c2ccc(O)cc2s1)c1ccc(N2CCCCCC2)cc1 C#CCC(C(=O)NCC(CC)CO)NC(c1cc(OC)n(C)n1)=O C(=O)(CCCC(C)(C)C)NC1CCN(C(c2ccc(CC)c(C)c2)=O)C(C)C1 C(=O)(C(CNC(=O)Cc1cc(C)on1)CC1CCCC1)NCC(CC)C c1(C(N(CCNC(=O)CC2CCCC2(F)F)CC)=O)cc(C)nnc1O C(CC(=O)N1CCC(CCO)(CO)C1)(C(C)OC)NC(CCOC)=O C=CCC(C(=O)N1CC(O)C(O)CO1)NC(c1ncncc1C)=O c1(CCC(=O)NCC(CNC(C23CCCC2C3(F)F)=O)OC)ccc(C)c(Cl)c1 Nc1cn[nH]c(=NCCS(=O)(=O)CC2CCC2)c1 CCCCC(C)C(=O)NC1CN(C(c2cccc(C3CC3)n2)=O)CC1C CC(CCNC(=O)CC1CCCOC1)CCNC(c1cc(=O)n(C)o1)=O c1(C(N2C(C)(C(=O)NCc3cnccn3)CCC2)=O)ccc2c(Br)cccc2n1 c1(C(N2CC(O)(Cc3nn[nH]n3)C2)=O)c(F)ccnc1F Cc1nn(C)c(C)c1CC(C)C(=O)NC(C)CC(C)NC(C1(C)C=CCCC1)=O Cc1nc(C)c(NC(=O)CCN(C(=O)CCNC(=O)OC2CCC2)C(C)C)[nH]1 C(=O)(N=c1[nH]nc(-c2ccc(C)cc2)s1)N(CCN(C(C)=O)C(C)C)C N1(C(c2sc(CC)c(C)c2)=O)CCC(O)(CNC(c2c(Cl)noc2C)=O)CC1 c1(C(N2C(CNC(CCC(=O)N(C)C)=O)CC2)=O)cc2c(F)cc(F)cc2[nH]1 C1(CNC(=O)COCC2CCCO2)CCC(NC(C2CCCC2)=O)C1 c1(C(N2CCC(NC(C(C#C)(C)C)=O)C(C)(C)C2)=O)cccc([N+](=O)[O-])c1OC N1(C(C2CCN(OC)CC2)=O)CCN(C(c2sc(N(C)C)nc2C)=O)CC(C)C1 C1(CN(C)C(C2CCC2)=O)CCCN(C(=O)C=Cc2sccc2Br)C1 CCCC(C)(O)CC(=O)N1CCC(CNC(C2CN3CCN2CC3)=O)C(O)C1 Cc1cccc([N+](=O)[O-])c1NCC(C)(C)C1(NC(=O)CC2CC3(CC3)C2)CC1 c1(OC)nc(N2CC3CCC(C2)N3c2ccnc(Br)n2)ncc1F C1(CCC(=O)NCC2CCC2NC(=O)Cc2ccccc2)CCCC(=O)N1 c1(-c2ccc(CN(CCCCCNCCC#C)C)s2)cc(CN(C)C)ccn1 c1(C(=O)NC2CC2NC(=O)C(O)Cc2ccc(F)cc2)cccc2ncccc12 c1(C(N2CC(CCC)N(C(=O)C(C3CC3)OCC)CC2)=O)c(C)cc(C)nc1S C(CC(C)N=c1nc(N2CCC3(CC2)NCCNC3=O)c2ncccc2[nH]1)SC C1(C)(CNC(C2C(C=C)OCC2)=O)CCN(C(c2nonc2CC)=O)CC1 CN1CC(NC(c2c[nH]nc2CCNC(=O)CN2C(=O)CCC2=O)=O)CCC1=O C1(c2n(CC(C)C)ccn2)CCCN(CC2(CCO)CCCC2)C1 C(=O)(CCCCCSC)N(CCCNC)C.C12(CC(=O)N(C)C)CCCC1C2 C#Cc1ccc(CC(=O)NC2CC(O)CN(C(=O)CCC3CCCC3)C2)cc1 c1(C(n2cc(C(C)NC(=O)C(c3cccc(F)c3)O)nn2)C)cccc(F)c1F C1(NC(C2N(CC)CC2)=O)COC2(CCN(C(=O)COCC(C)(C)C)C2)C1 c1(C(N2CCC(CNC(c3ccc(F)cc3)=O)C23CC3)=O)ccc2c(n1)CCO2 c1(C(=O)NC2CCN(C(C3(O)CC(C)(C)C3)=O)C2)cc(C(=O)CBr)ccc1O C1(C(CNC(c2c(C)ocn2)=O)F)CCN(C(c2c[nH]ccc2=O)=O)CC1 Cc1cc(C(=O)NC2CCN(C(=O)C(=O)NC3CC3)CC2C)c2c(O)n[nH]c2n1 N1(CC)CC(C(N2CCC(CNC(C3CC(C)=NO3)=O)C2)=O)CCC1=O Cc1nsc(C)c1C(=O)NCC1C(C)CCN1C(=O)Cn1cncn1 C1(C(=O)NC(CC)CC(=O)NC2CCCCCC2)CCC2(CC2)CO1 c1(C(=O)NC(C2CCN(C(=O)CC3NC(=O)NC3=O)C2)C)nnn2c1CCC2 c1(CNC(c2c(CC)scc2)=O)ncccc1CNC(=O)C(C1CCCO1)OC C(=O)(C(F)C(C)(F)F)NCC(C)(CO)OC.C12CC13CC(C3)NC2=O N1(C(CCC(C)SC)=O)CCC2(CC1)CCN(C(c1cn3cc(C)sc3n1)=O)C2 [N-]=[N+]=Nc1ccnc(NC(C2CC2C(N2C(CNN)CC2)=O)=O)c1.C(=O)NCCNC(N)=O c1(C(CCOC)NC(=O)CC2CNCC2O)ccccc1Cl C1(C(=O)NCC(C2CCC2)NC(c2cncc(C)n2)=O)CCC(F)(F)CC1 N1(C(c2cc(C)sc2C)=O)CC2CC1CN2C(=O)C(C)(O)c1ccccc1 C1(C(=O)Nc2c(OCC)scc2)CCN(C(=O)CC2(C)CCCO2)CC1C C1(C(=O)NC(COC)CCO)CC(C)(C)CCN1C(C1CCC(C)(C)C1)=O Cc1cc(C(=O)NCC2(NC(C3CC(C)CC(C)C3)=O)CCCC2)cc(C)c1Cl C(CCCN=c1[nH]c2ccc(C(=O)OC)cc2s1)OC.c12sccc1C(=O)NC2 c1(CC)ccc(C(=O)NCCCCCCNC(C2CC2(F)Cl)=O)cc1Br Cc1cc(C)c(OCC(=O)NC(C)CN(C)C(C2(C)CCN(C)C2=O)=O)c(C)c1 C1(COC)CC(CNC(=O)CCc2cc[nH]n2)N(C(c2cc(C(F)F)[nH]n2)=O)C1 Cc1csnc1C(=O)NCCC1CC(NC(=O)CCC2(C)CC2)C1 C1(C(N(CC=C)CC)=O)CC=CCN1C(=O)C(C)CCOC C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(=O)N(C)C)C2(CCCOC2)C1 C(C(C)C)(C(O)C(=O)NCC(C)(C)NC(c1cc(Cl)cnc1O)=O)OC c1(C(=O)NC2CC(CNC(c3cc(CCC)on3)=O)CC2O)ncc(N)cc1Cl c1(C(N2CCC(OC)(CNC(c3cncnc3C)=O)C2)=O)cnc(Cl)c(Cl)c1 C1(F)(CNC(C)=O)CCN(C(=O)C(c2cccc(C#N)c2)C)CC1 C1(CC(=O)Nc2nnc(C3CCN(C(CCC#C)=O)CC3)s2)CCOCC1(C)C O=C(C1CCCc2nccn21)NCC1CC12CCN(C(=O)CC=CC)CC2.C c1(C(=O)NC(C)CCCCNC(=O)CC(F)F)ccc(Cl)c(Cl)c1N c1(OC)ccc(CNC(=O)CC2CSCCS2)cc1OC c1(NC(=O)Nc2c(NC(=O)OCC)c(C)ccc2)cnc2cc(F)ccc2c1 Cc1csc(=NCC(=O)NCC(C)(C)CNC(c2cc[nH]n2)=O)[nH]1 C(C(=O)NCc1cccc(CNC(=O)CCOC2CCCCC2)c1)(C(C)C)SC C1(C(=O)NCC2N(C(C34CC3C4)=O)CC=C2)CCCCC12CCC2 c1(CC)ccc(F)cc1C(=O)NCC=C1CCN(C(=O)C(C)C(C)CC)CC1 C(=O)(C1CCCCc2ccccc21)N(C)CC1(O)CN(C(c2cc(C)no2)=O)C1 c1(C(=O)NCC2CCCN(C(C(c3c(C)noc3C)C)=O)C2)cccc(N)c1C C1(C(=O)NCC(C)N(C)C(c2cc[nH]n2)=O)CN2CCCC1C2 N1(C(C2C(=C)CC2)=O)CC2CC2(CNC(c2cncc(C(F)F)c2)=O)C1 c1(OC)ccc(CN(C(c2cc(Br)ccc2F)C(=O)NCC2CC2)C)c(F)c1F Cc1cc2ccc(C(=O)NC(CO)CCCCNC(=O)CCC3CC3C)cn2c1 c1(CC)oc(C(=O)NC2CC(CCNC(=O)C(c3ccccc3)C)C2)cc1C c1(C(=O)NC2CCN(Cc3ncc(Br)s3)C2)cc(O)ncn1 C(CCCCC(=O)NC(C)CS(C)(=O)=O)N(C(c1cc(CC)oc1C)=O)C c1(OC)cc(C(N2CCC(NC(c3ncc(F)cc3C)=O)C(C)C2)=O)cc(Cl)n1 C(C(COC)C(=O)N(C)CC1CCCC(NC(c2ccn(C)n2)=O)C1)OC c1(C(=O)OCc2c(C)non2)cccc2cccnc12 C1(NC(CNC(CC)=O)=O)CCC(CCNC(c2nc(C(C)(F)F)cs2)=O)C1 C(CCC(=O)NC(C)CNC(C1CC(F)(F)C1)=O)NC(=O)OCC N1(C(C(C)NS(C)(=O)=O)=O)CCC(C2(C(=O)NCC(N)=O)CCOCC2)CC1 N(C(=NCCC(C)=O)NCC1CCCO1)C1N(CC)CCC1.c1cc(F)cc(F)c1 C1(NC(C(C)n2cnnn2)=O)CCC(O)CN(C(=O)C=CC(F)(F)F)C1 N1(C(c2cc(C)nc(O)n2)=O)CC2CC1CCC2NC(c1n[nH]cc1Br)=O CC(C)C(C(=O)NCC(C)(C)CN(C(=O)C(O)C1CCC1)C)N(C)C c1(C(C)(F)F)cncc(C(=O)NC2COCC2NC(c2c[nH]c(=N)s2)=O)c1 N1(C(C(C)OCCC(C)C)=O)CCC(NC(=O)C2=CC(C)(C)C2)C2(CCC2)C1 C(=O)(C(F)(CNC(=O)COCCCC1CCC1)C(C)C)NCC(C#C)C.N(C)C N1(C(CC2ON=C(C)C2)=O)CC2CC(O)C1C2NC(c1cccc(Cl)c1O)=O c1(C(N(C2CCC(C)CC2)C)=O)n[nH]c2c1CN(C(C1(C)CCCS1)=O)C2 N1(N2C(C(=O)Nc3ccc(Br)cc3CC#N)CC3CC32)Cc2ccc(F)cc2C1 c1(C(N2C(CNC(c3c(OC)scc3)=O)CC2)=O)ccccc1C(=O)N(C)C c1(C(=O)NCC(CC)NC(C2CCCCC2(F)F)=O)cc(Br)c2occc2c1 c1(C(N2CCC(CC(C)NC(C(CC)SC)=O)CC2)=O)cc(N)c(Cl)cn1 n1(C(C)C(=O)N(C2CCOCC2)C)cnc2ccccc12 N1(C(C(CC(C)C)OC)=O)C2CCC1CC(CNC(c1cc(C(F)F)no1)=O)C2 C(=O)(C(CCOCCO)NC(=O)CNC(N)=O)NCC(CC)(C)Cl CC1CN(C(C2CC(F)(F)C2)=O)CCN1C(=O)C(F)(F)C1CCOCC1 N1(C(Cc2c(C)occ2)=O)CCC(NC(=O)C=C2CCC(C)C2)C1(C)C CC(C)C1=NOC(CNC(=O)NCCCC2CC3C=CC2C3)C1 c1(N(C(=O)COc2ccc(F)cc2C(N)=O)C)ccc2c(c1)CCC2 C1(CC(=O)N(C)Cc2cccs2)CCN(C(c2ccccc2)=O)C1 C1(CNC(CC2CC(C)C2)=O)(CNC(=O)CC2OCCCO2)CCCC1 CC(C)CC(C)CC(=O)NCC(C)(C)CCNC(=O)C=CC=C(Cl)Cl C1(C(=O)NCC2CC(NC(c3cnn(CCCC)c3C)=O)C2)CCC(C)(C)CO1 CC(C(=O)NC(C)(CNC(=O)CCOc1ccccc1)C1CCC1)P(C)(C)=O C1(NC(c2ccc(C)cc2O)=O)CC2CC1CN(C(=O)C=Cc1c[nH]nc1C)C2 CCC(CC(=O)NCC1CN(C(c2ccsc2C#N)=O)CCC1(C)C)C(F)F C12(C(N3C(C(=O)NC4(C)CCSC4)CC(O)C3)=O)CCC(CC1)CC2 C(c1cccc2ccccc12)=CC(=O)NC1CN(C(c2c(C)occ2)=O)C2C1C2 c1(SCC(=O)NC2CCC2NC(=O)Cn2cncn2)ccc(Cl)nc1 N1(C(C(CCC)OC)=O)CCCC(NC(c2cnn(CCN(C)C)c2C)=O)C1C C1(NC(Cc2c(C)noc2Cl)=O)CCC2CN(C(=O)C(F)F)CCC2C1 S(=O)(=O)(CCC(=O)NC(CNC(=O)CN1CC=CC1)C1CC1)NC CS(=O)(=O)CC(=O)N(CCC(=O)NCC1CCCC12CC2)CCO Cc1nnc2n1CCC(C(=O)NCCC1(NC(c3cc[nH]n3)=O)CC1)C2 n1(CC)ccc(S(=O)(=O)N2CCC3CCC23C(=O)Nc2cccc(CO)c2)n1 c1(CN2C(C)(C(=O)NCCCC)CC2)ccnc(Br)c1F C1(C(=O)NC(C(N)=O)C2CC2)CCC(C2CC2)N1C(c1c[nH]c(=O)cn1)=O CCC(C(=O)N1CC(O)(C2CCCN2C(=O)CSCc2ccncc2)C1)SC c1(OC)cc(C#N)ccc1-c1noc(-c2cc3scnc3[nH]2)n1 C1(C(=O)NCC2(C(C)(F)F)CCC2)CCC(CNC(=O)C(F)C2CCCC2)O1 C(C)(C)(CC(=O)NC(C1CCCN1C(=O)CC1(N2CCCC2=O)CC1)(C)C)OC N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CCC(NC(=O)C(C)(C)OC)CC2)C1 N1(C(CC2(OC)CCC2)=O)CCN(C(c2nn(C)cc2N)=O)C(C)C1 CC(C)C(C(=O)NCCC(C)N1CCCC1)C(C)NC(C1(C)CCCC1)=O C=Cc1ccc(N(C=O)CCO)cc1.C1(SC)CC2(CC(=O)C2)C1 C(C(C)(C)C(=O)NCC1CCCN1C(c1cnn(C(F)F)c1)=O)OCC CCCCC(CNC(=O)Cc1cccnc1C)NC(C1(C)CCC(=O)N1)=O CC(CC(=O)Nc1cccc2c1OCO2)C(C)(C)NC(=O)C=CCN1CCCC1 c1(C(=O)NC(C)C(CO)NC(c2ccnn2CC(F)(F)F)=O)ccc(F)c(F)c1 C1(O)(CC(=O)NCC(CNC(C(n2cc(C)nc2)(C)C)=O)O)CCCN(C)C1 c1(CNC2CCC(C(=O)Nc3ccc(Cl)nc3)C2)cc(F)ccc1NCCCC C1(C#CC(=O)N2CCC(N(C(=O)CC(C)(C)O)CC3CC3)CC2)(CC)CC1 c1(C(=O)NCCCN(C(C2CCC(=O)O2)=O)C2CC2)cccc(-n2ccnc2)c1 c1(OC)ccc(SC(C(=O)O)C(=O)O)cn1.C1C(CCN(C)C)N1 c1(C(=O)NCc2ccc(CNC(C(CC)COC)=O)cc2)ccc(Cl)c(C)c1 C(=O)(C(=O)N=c1ccn(C(c2ncccn2)C)[nH]1)OC.n12ncnc1C(C)(C)C2 C(CN=c1ncc(C(F)F)c[nH]1)C1CCN(C(=O)CC2C=CCC2)C1 c1(NC(c2ccccc2)COC)[nH]c(=NC2CCCCCCC2)nc2scnc12 c1(C(=O)NC(C(C)O)C(N)=O)cc(-c2cccc(CN3CCCC3)c2)cnc1F N1(C(c2c(CNC(C=CC=CC)=O)oc(C)c2)=O)CCC(OC)C(C)(C)C1 c1(C(=O)NC(CNC(C2CCCN2C2CC2)=O)CO)cc(F)cc2ccncc12 C(C)(C)(C(C)CC(=O)NC(C)C(C(=O)O)C(C)C)NC(c1ccc(C)c(C)c1)=O n1(CC(=O)NC(C)CCCNC(c2ccon2)=O)cc(C#N)c(O)nc1=O C(CC1=CCN(C(C2CC23CCCCC3)=O)CC1)NC(c1cc(C(N)=O)[nH]c1)=O C1(OC)CC2CC(NC(=O)C(C)(C3CC3)NC(c3nnsc3C)=O)CC12 C1(CCN(C(C(F)=CCC)=O)C)CCCCN1C(=O)CC1CCC(=O)N1C c1(CC(=O)NC2CCCN(C(C3CCO3)=O)C2)c[nH]c2ccc(Br)cc12 C1(NC(c2scc(CC)c2)=O)CCCCC12CCN(C(c1cc(C#N)on1)=O)C2 c1(C(=O)NC2(C)CC(NC(C3CC(=C)C3)=O)C2)noc2c1CCCC2 C1(NC(C(C2CC(NC(C(C)OCOC)=O)C2)F)=O)CCc2n[nH]cc2C1 C1(C(C)(C)NC(C(CC)NC(C)=O)=O)CCCCN1C(c1cn(C2CC2)cn1)=O C1(C(=O)NC(C(N)=O)CO)(NC(c2ncncc2Cl)=O)CC(F)(F)C1 CCCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(c1[nH]nc([N+](=O)[O-])c1Cl)=O Cc1ccccc1-c1nc(C(=O)NCCN(C(=O)COC(F)(F)F)C)cs1 c1(CCC(=O)NCC(CC)NC(COC(CC)CC)=O)nc(C)c(C)[nH]1 c1(C(=O)NC2(C)CN(C(c3c(COC)cco3)=O)C2)ncn2c1COCC2 C1(C2CCOCC2)(C(N2C(CNC(c3c(C)nc(CO)o3)=O)CC2)=O)CC1(F)F C(=O)(C1CCc2ccccc21)N1C(C=CC(=O)NCC2C(=O)OCC2)CCC1 C1(NC(C2CCCSC2)=O)CCC2(CC1)CN(C(C1CN3CCN1CC3)=O)C2 c1(CCC(=O)NC(CC=C)CNC(=O)C(C)O)cc(OC)ccc1OC Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NC1CCCCC1NC(=O)C1=CCCOC1 c1(C(=O)NC2C(CNC(c3cc(OC)c(F)cc3)=O)C2)c(C)nc2sc(C)cn12 CC1CCC(C)(C(N2CC(CN(C(=O)CCCC#N)C)C2)=O)C1 C1(C)(CC)CN(C(C(=O)Nc2ccccc2OC)C2CCOC2)CCO1 c1(CC)ncc(C(=O)NC23CC(C(N4CCC4CO)=O)(C2)C3)cn1 N1(C(C(C)NC(CC)=O)=O)CCCC12CCN(C(=O)C#CC1CCCCC1)C2 N12CCC3(CC1)CC3N(CC)C(CC=C)C2=O.C1(=CC(=O)NC)CCC(C)C1 CC(C)C(F)C(=O)NCCC1CC(NC(c2csc(Br)c2Cl)=O)C1 N1(C(C(C)(C)C2CC(C(N3CCCCC3)=O)C2)=O)CCN(C(=O)CCCC2CC2)CC1 C1(CNC(CCSCC)=O)(NC(=O)CN2CCCCC2C)CCCCC1 c1(C(N(C2CCN(C(C3C(C)C3C)=O)C2)CC)=O)cc(F)c(C)cc1Cl N1(C(c2ccc(C)cn2)=O)CCCC2(CCC2NC(=O)CC=C(Cl)Cl)C1 C1(C(=O)NCC2(NC(CC3(C)CC3)=O)CCC2)CC(=O)CO1 c1(OC(C)C)nc(C(N2CC(CCNC(=O)COCP(C)(C)=O)C2)=O)cc(O)n1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)CC2C)csc2c(F)cccc12 C1(C#CC(=O)NC2CC(O)(CNC(=O)C3=CCCCC3)C2)(CC)CC1 N1(C(c2cc(C)n(C)c2)=O)CC2CCC(C1)N2C(=O)CSC1CCS(=O)(=O)C1 c1(C(N2CCN(Cc3ccccc3)C(C3CC3)C2)=O)cc(Cl)c(F)cc1F N1(C(=O)CC2C=CCC2)CCC2CN(C(c3cc4c(nn3)CCC4)=O)C2C1 c1(N(C(CC(CC)NC(C23CC(C)(CO2)C3)=O)=O)C)cc(C)ccc1C c1(C(=O)NCC(CNC(c2n(CC)ccn2)=O)CO)ccc2ccsc2c1 C(=O)(C(CC)C(=O)NC1CC(F)(CNC(=O)C(C(C)C)SC)C1)OCC C=C1CC(C(=O)NC2CN(C(C)=O)C2)(C(C)N)C1.C1(C)CCC1C(C(=O)OCC)=O C1(C(=O)NCCC2(C)CCN(C(COCCC)=O)C2)CC2CCC(C1)O2 Cc1cnc(NCC(C)(C)C2CC2)c(S(=O)(=O)N2CCC(OCCCO)CC2)c1 c1(C(c2n(CC(=O)OC)nnn2)NCC=Cc2cccs2)ccc(OC)c(C)c1 n1(CC)ccc2cc(C(=O)N(C3CCN(C(=O)C4CC4)CC3)C)ccc12 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC2(C(NC(CCCC#CC)=O)CC2)C1 Cc1cccc(-c2cnccc2C(=O)NCCC23CC2CCN3)c1.C(=O)OCC C12(C(=O)NC3CNC(=O)O3)CCCC1CN(Cc1ccc3c(c1)COC3)C2 c1(CC(=O)NC2CC(NC(C3C(C)OC(C)C3)=O)C2)csc2ccc(Cl)cc12 CC1(C)OCCOC1C(=O)NCCC1CCCCN1C(c1ccc(Cl)cc1)=O C1(NC(C(C)=C2CCCC2)=O)C=CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(CC(=O)NC2CN(C(C3CC3COC(C)(C)C)=O)C2)c[nH]ccc1=O N1(C(C2ON=C(C(C)(C)C)C2)=O)CCOC2CN(C(c3nc(Cl)cs3)=O)CC12 C(C(C)CC(=O)NNC(=O)C(C)(C)CCCCSC)NC(=O)CN=S(C)(C)=O.CO c1(C(=O)NC2C(CNC(=O)CCCc3ccsc3)C2)ccc2n[nH]cc2c1Cl c1(OC)ccccc1NC(=O)C(C)N(C1CCN(CC2CC2)CC1)C C1(CC(N2CC3C(NC(C4C(OC)CCC4)=O)C3C2)=O)CN2CCN1CC2 N1(C(c2cc(C)n(C)c2)=O)CCC(C(=O)NCCC2CCOC2)C(C)C1 C(C)(C(CC(=O)N(CC)OC)NC(C1CC(C(=O)OC)C1)=O)OC C1(C(F)(F)F)(C(=O)NCCC2(NC(C=C(C)Cl)=O)CCCC2)CCCCO1 C1(NC(CN(CCCCCC)C)=O)CC(CO)N(C(=O)CC(C)n2cccn2)C1 c1(OCC)ccccc1CCC(=O)NCC1CC(NC(C2CC(F)C2)=O)CC1O Cc1c(C(=O)NC2(CCCNC(C3(C)COCCO3)=O)CC2)ccn1C N1(C(=O)NCC(N2CCNC2=O)(C)C)CCC(CO)CC1(O)C C1(C(=O)OC)CCOC1C(=O)NC12CC(NC(=O)CCSc3ccccn3)(C1)C2 c1(NCC(CC)(C)OC)cc(N(C)Cc2ccc(=N)[nH]c2)ncn1 CC1CCCCC1CC(=O)N(CC(O)CN(C(=O)CN(C1CCSC1)C)C)C CC1CCN(C(=O)C=CC=C(Cl)Cl)CCN1C(=O)COc1cncc(O)c1 c1(C(N(C2CCN(C(C=CCCC)=O)C2)CC)=O)ccc(=O)n(O)c1 N1(C(CCC#C)=O)CCC2(CC2NC(=O)CCNC(c2ccccc2)=O)C1 N1(C(c2nc(OC)c(F)cn2)=O)CC2=C(C1)CN(C(=O)C(C1CC1)SC)C2 C1(C(=O)OC)CCC(C2(C(=O)OC(C(=O)NC(C)C)(C)C)CCC2)CC1 C1(CC)CN(C(C2(NC(c3cc(C(C)=O)c[nH]3)=O)CCC(C)(C)C2)=O)CCCO1 c1(OC)c(Cl)cc(C(=O)NC2CCCN(C(=O)CN3CCC3C)C2)nc1Cl C1(C(=O)NC(C)C(C)O)(COC)CN(C(=O)CN(C)C2CC2)C1 c1(C(=O)NC2(C)CN(C(C3(C)CCCC3)=O)C2)ccc([N+](=O)[O-])cc1Cl C1(CC(=O)NCC(=O)OCCCC)CN(C(c2ccc(C)[nH]2)=O)CCC1C c1(CNC(CC=C=C)=O)cccc(C(=O)NCCCN2CCCC2=O)n1 C#CCCCC(C(=O)NC(C)(C)CC)N1CCC(OCCN(C)C)C1 c1(NCCNC(c2ccc(Br)cc2)CC)ccc2c(c1)CCCN2C N1(C(c2cc(CCC)on2)=O)CCOC(CNC(=O)CCCCN2CCCC2)C1 Cc1nc(NC2CCCc3c[nH]c(=N)nc32)c(Cl)cc1C#N.C1(C)C(=O)N1 N(C1CCc2ccc(Br)cc21)C(CCc1ccc(OC)cc1F)=O C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(c2cocn2)=O)C1 c1(CN2CCC(NCC3(C(=O)OCC)CCC3)C2)ccccc1C C1(O)(CN(C(=O)CCOc2cccnc2)C)CCCN(C(=O)CC2OCCO2)C1 N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CC2)(C(=O)NC(C)C(O)C(F)F)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C)CCN(C(C(COC)C)=O)C1 c1(CNC(C2CCCCN2Cc2c(F)cccc2F)=O)c(F)c(F)cc(F)c1F C(=O)(C(CCC1CCC1)NC(=O)CC1C=CCCC1)NC(c1cc(C)on1)C C1(NC(C(C2CCC2)OC)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 c1(CC(=O)NC2C(NC(CCN(CC)CC)=O)C2)c[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)N1CCCC(CC(N2CC(OC(=O)NC)C2)=O)CC1 C1(NC(=O)CO)COCCN(C(C2CC(=O)NC2(C)C)=O)C1.C1(=O)CCN1C C1(C(N(CC(c2ccccc2)O)C)=O)CC2CC(C1)N(C(c1cc(O)no1)=O)C2 c1(C(=O)NC2CN(C(C=CC(=O)OCC)=O)CC2O)cc2scc(Cl)c2[nH]1 c1(C(=O)NCC(CO)NC(c2c(C(C)(C)C)con2)=O)ccc(F)c(Cl)c1F C1(c2nc(-c3ccc(OC)cc3)nn2CCNS(N)(=O)=O)CCC2(C1)CC2(F)F c1(C2N(c3nnc(CC(CC)C)n3CC)CCC2)cc(OC(F)(F)F)cc(F)c1 C1(NC(C2(OC)CCSCC2)=O)CCN(C(=O)CC2CCC3CC23)CC1(C)C CC(C)(C(=O)N1CC2CC1CC2CNC(=O)C(C)(C)C1CCCO1)C(F)F CN(C1CCc2c(F)cccc21)C(=O)CC1CCCC1(F)F C1(NC(CC)(CC)CO)CC(C)(C)CCC1=O C=C(C)CC(C(=O)NC1CS(=O)(=O)CC1NC(c1sc(C)nc1C)=O)OC CC(C)C(F)(CNC(C1C2CC(=O)CC12)=O)C(=O)NCc1cccnc1O c1(C(N2CC(C)(C)C(NC(C3CC(C#N)C3)=O)C2)=O)cc2cc(Br)cn2cn1 C1(NC(C(C)OC)=O)CN(C(c2c(C)nc(C)n2O)=O)CC2(CCC2)C1 C1(C(=O)NC(C)CCCNC(C2CC2c2cc[nH]c2)=O)CCCN(c2cccs2)C1 C(=O)(C1=CCSC1)N1C(C)(CC(N2CC(C(C)OC)C2)=O)CC1 N1(N2C(C)(C(N3C(C=O)CCC3C)=O)CC2)CCc2ccncc21.CS C1(O)(CCNC(C2CC(=O)NC2)=O)CCCN(C(c2cncc(O)c2)=O)C1 CCC(CC(=O)N(C1CC(C(=O)NCC2(C3CC3)CCCO2)C1)C)OC C1(NC(c2n(CC)ncc2)=O)CCC(C)(CNC(c2cnc(C(C)O)s2)=O)C1 C1(NC(CC(C)(C)C)=O)CCC(C)(NC(c2ccoc2Cl)=O)CC1 CCCC(CCC)CC(=O)NC1CC(OCC(N2CCCC2C(=O)NC)=O)C1 c1(OC)cc(C(=O)Nc2cnc(Cl)c(CO)c2)c(-c2cncn2C)cn1 N1(C(c2cnn(CC)c2Cl)=O)CC(NC(C2CC(C(N)=O)C2)=O)CC(F)C1 C1(C(N(C2(C(=O)NCCS(C)(=N)=O)CC2)C)=O)CCCC1C1CC1 N(C1CCc2cccc(Br)c21)CCn1ccc2c(NC(C#C)(C)CC)ncnc12 N1(C(C(C)OCCOC)=O)CCCN(C)CC1C.C1C(C)(C)C(=O)N(C)CCO1 c1(NC(=O)CC(F)(F)F)nncc2c1CCCC2.CC1(C)C2CC1CNC2=O C1(CNC(C(c2cccs2)SC)=O)CCCN(C(=O)C=Cc2ccsc2)C1 C(=O)(CCCC(O)C1CSC1)N(C(C)COC1CCOC1)CCC C(=O)(CC(C)(C)C(F)F)N1CC(N(C)C(C2C(=O)NCC2(C)C)=O)C(O)C1 C(C(C)CC(=O)NC1CCCN(CCC)C1)NC(CN(CCC#C)C)=O c1(OC)cc(O)c(CN2CC3C(C2)N3C(c2ccc(Br)s2)=O)cc1Cl c1(CCC=C)ccc(C(N2CC(CO)(NC(C3CN(C)CCO3)=O)C2)=O)cc1 c1(CCCC(=O)NC2CCN(C(CCC(=O)NC)=O)C2C)ccc(OC)cc1F C(=O)(C1CCCc2nn(C)cc21)NCC1(NC(c2nn(CC)c(O)c2)=O)CCC1 CC12CN(C(=O)CN3CCOC3=O)C(C(CC=CC(=O)OC(C)(C)C)=O)(C1)C2 c1(C(=O)NC(C)CC(=O)NCCC2CCCC2)cc([N+](=O)[O-])c[nH]1 N1(C(=O)Nc2cc(N3CCN(C)CC3)ncc2)CCC(C)(O)C(C)(O)C1 Cc1ccc(Br)c(CNC(=O)NCC(C)(C)NC(N)=O)c1 N1(C(c2n(CC)ncn2)=O)CCCC(C2CCN(C(c3cnnc(Cl)c3)=O)C2)C1 C1(NC(c2csnc2C2CC2)=O)CN(C(=O)CC2=CCCCC2)CC2(CC2)C1 C(=O)(C(C)(C)C(C)(F)F)NC(C(=O)NC(COCC)C(C)C)COCC C1(NC(c2cc(C)c(Br)o2)=O)C2CC1CN(C(C1CCSCC1)=O)C2 c1(C(=O)OC)csc(C(N2CC(C)C(F)C2)C(=O)NCCCSC)c1Cl Cc1ccccc1CC(C)C(=O)NCC#CCNC(C1(C(=O)NC2CC2)CC1)=O C1(NC(CSC)=O)CCN(C(c2nc(-c3ccccc3)oc2C(C)C)=O)C(C)C1 C1(NC(c2nc(COC)sc2)=O)CC2CN(C(=O)C(F)C3CCOC3)CC12 CCCC(CNC(=O)CCc1csnn1)NC(C1CCN1C)=O C(=O)(CCCCCC(C)O)NC1COCCN(C(c2ccc(C)c(C)c2)=O)C1 Cc1ncc(CNC(=O)C(C)CN(C(=O)C(=C2CCCCC2)F)C)o1 c1(OC)cc(NCC2CCCCC2NC(=O)C(F)CC2CCCCC2)ncn1 N1(C(CC2CCCC(NC(C=CC(CC)C)=O)C2)=O)CCCC2(CCC2)C1 C1(C(=O)NC2C(SC)CN(C(=O)Cc3cncs3)C2)CC12CCC1(CC1)CC2 C1(NC(c2ccc(OC)s2)=O)CC(NC(=O)C=CSC)C12CCC2 Nc1c(C(N2CCC(NC(=O)Cn3cnc4ccccc34)C2)=O)cc(F)cc1Cl C12(N(C(c3ncccn3)=O)CC3(NCc4ccccc4)CC3)CC(F)(C1)C2 c1(C(N2CC(CCC)N(C(c3cnn(C)n3)=O)CC2)=O)ccc2snnc2c1 CCC(C)CCCCC(=O)NCC1CCC2(CN(C(=O)OC(C)(C)C)C2)OC1 C=CC1CCN(C(=O)CC2CC(F)CN2C(=O)C(C)NC(=O)NC)C1 C=CCCCCC(=O)N(CC(CC)NC(=O)COc1ccccc1C(C)C)C C1(C(N2CC(NC(C(C)OC3CCCC3)=O)C(O)C2)=O)CSc2ccccc2O1 C1(CNC(CCSC)=O)CN(C(=O)CC(C)n2cccc2)CC(C)(C)C1 C1(C(N(C2CN(C(c3cccc(OCC(F)(F)F)c3)=O)C2)C)=O)CCC(C)(C)C1 CC(C)CC(C(=O)NC(C)C(=O)NOC1CCC(O)C1O)C(N)=O n1(CC)ncc(Br)c1-c1nc(-c2ccc(Cl)nc2)nn1C(C)C(C)C C#Cc1ccc(Br)c(C(=O)NCC(C2CC2)NC(C2CCN(C)S2(=O)=O)=O)c1 C1(CC=C)(NC(=O)CCS(C)=O)CCCN(C(C2CC2(c2ccccc2)C)=O)C1 C(=O)(N=c1cc[nH]cc1F)C1(C)CCN1NC(c1cccc(I)c1)c1ccccc1 N1(C(CC(C)C(F)F)=O)CC(CNC(c2cn3c(n2)CCC3)=O)CC12CCC2 c1(C(N2CC(O)(CCNC(=O)CO)C2)=O)c(Cl)nsc1Cl CCCC(C)(O)CNC(C1(CCNC(=O)Cc2coc(C)n2)CCC1)=O c1(N2C(CNC(c3csc(C4CC4)n3)=O)CC(OC)C2)ncc(C#N)cc1Cl c1(C(N2CC(NC(CCC(C)C)=O)C(C3CC3)C2)=O)ccc2c(c1)C(=O)NCC2 N1(C(CC2(C)CCCC2)=O)CCCC(C)(CNC(C2CC23CCCC3)=O)C1 c1(C(N2CC(NC(CC(C)n3cccn3)=O)CC2(C)C)=O)ccc2occc2c1 c1(C(N(C(C)CNC(C2CCCN(C(=O)OC)C2)=O)CC)=O)c(N)ccc(C)c1F NC(=O)CCCCC(=O)N(CCCNC(C1CCC(C(=O)OC)CC1)=O)CCO N1(C(CC(C)(F)F)=O)CCC2CCC(C1)N2C(C1CCc2cncn2C1)=O S(=O)(=O)(c1c[nH]ccc1=NCCC1CCCC1O)NCCN=S(C)(C)=O Cc1cnc(C(N2CC(F)CC2CC(=O)NCC(C)(O)C2CC2)=O)c[n+]1[O-] c1(CNC(C23C(CN(C(c4ccc(Cl)o4)=O)C2)C3)=O)cnc2n1CCC2 C(=O)(C(C)CC1CC1)NCCC1CN(C(CNC(C)=O)=O)C1 C1(C)(C(=O)NC(CC)CNC(=O)Cn2ccnc2C(C)C)CCSCC1 CN1CCCC12CCN(c1nccc(=NCCOC(F)F)[nH]1)C2 C(=O)(C1=NOC(C)(C)C1)NC1C(C(=O)NCC2C(C)OCC2)CCC1 n1(CC(=O)NC2C(NC(C3(C)CCC3)=O)CCC2)cc([N+](=O)[O-])cn1 N1(C(C2=CC(C)(C)C2)=O)CCC(NC(C2CC(F)(F)C2)=O)C12CCCC2 c1(C(N2CCC(O)(CNC(CSC)=O)C2)=O)ccc2cnccc2n1 C(=O)(CCCCCS(N)(=O)=O)N1CCN(C(CC2=C=CC(N)=C2C)=O)CC1 CC(C)CCCC(=O)N1CCCC1CC(=O)N(CCO)CC1CC1 C=C(F)C1(CC(=O)NCC2CCC(NC(=O)C(F)=C(C)C)CC2)CCC1 CC(CN(C)C)C(=O)NCCCOCCC(=O)NCC1CSCCO1 N1(C(c2n(C)c(S)nn2)=O)CCCC2(C1)CN(C(=O)CN1CC(C)(C)C1)CCO2 C1(C(=O)NC(C=C)COC)CCCN(CC2CCC2)C1 C1(NC(C2CCC(C)O2)=O)COC2(C1)CN(C(c1cc(Cl)on1)=O)C2 C(=O)(C(O)C(F)(F)F)N1CCC(N2CCN(C(C3(C#N)CCCO3)=O)CC2)CC1 c1(C(N(CC(C)O)CCNC(C2(C(C)C)CCC2)=O)=O)cncc2cccnc12 CC(C)(C)CC(O)C(=O)NCC1(F)CC(NC(=O)CC2CCCC2(F)F)C1 C1(=O)C(CC(C)C)NC(=O)CC2CC(C)N1C2.c1(CC)onc(C)c1CN CC1CN(C(=O)CN(C)C2CC2)CC(C)C1NC(c1cc2sccc2s1)=O Nc1ccc(-c2noc(Cc3cnc(-c4ccccc4)o3)n2)c([N+](=O)[O-])c1 c1(C(=O)NC(CNC(CCOC)=O)(C)C(C)C)cc2c(C)cccn2n1 CCC(C)(C)CCCC(=O)NCC(CNc1cc(C)nc(SC)n1)C(F)(F)F N1(C(CCNC(c2ccc(F)cc2)=O)=O)CC2CC(O)CC(C2)C1 C(CCC(C)CC(=O)NCCC1CSCCN1C(=O)CCS(C)(=O)=O)=C(C)C C(=O)(CCC(CF)CF)N1CCCCC(C(N(C)Cc2cncnc2)=O)C1 c1(C(N2C(C(=O)NCc3c(C)cco3)CCC(O)C2)=O)ccc2cccnn12 C1(OCC(=O)NC2CC(NC(C(=O)N(C)C)=O)CC2O)CCC(=O)NC1=O C(N(C)N1CCN(S(C)(=O)=O)C2(CCCC2)C1)c1cn(CC)c2c1cccc2 C(CC(C)C)(C(=O)OCC(C)(C)C)OC(C)=O.C(C)CN(C)C(C)C CCCC(C(O)C(=O)NCCN(C(C)C)C(C)C)NC(=O)C(F)OC(F)(F)F C=CCC(C)(C)C(=O)NCCC1(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1 c1(OC)ccc(S(=O)(=O)N(c2ccn3nccc3n2)C2(SC)CCNCC2)cn1 c1(C(=O)NC(C2(O)CN(C(c3c(C)nsc3N)=O)C2)C)csc2cc(Cl)cnc12 C1(N(c2cnn(C)c2)CC)CCCN(C(=O)C(N)=O)CC1 c1(C(N2C(CNC(=O)Cc3ccc(F)cc3C3CC3)CC2)=O)n[nH]c2c1COCC2 C1(C(=O)OC)CC2(CCCC2)CN1C(c1cc(Cl)cc([N+](=O)[O-])c1N)=O C12(CNC(c3ccc[nH]3)=O)CC(C1)C(NC(C1CCCC(F)(F)C1)=O)CO2 CCC(N=c1cc(C)c(C#N)c(C)[nH]1)C1CCCCN1C(C1CC=C(C)CC1)=O CN1CCC(=CC(=O)NCCC(O)CNC(c2ccccc2CO)=O)CC1 CCCS(=O)(=O)C(C)C(=O)N1CCCCC1CN(C(=O)CSc1cccs1)C N1(C(COc2ccn(C)n2)=O)CC(NC(c2scnc2C(C)(C)C)=O)CC(O)C1 c1(NC(C2NCCN(S(CC#N)(=O)=O)C2)=O)ccc(F)cc1[N+](=O)[O-] CC1S(=O)(=O)CC1CCC(N1CCCCC1Cc1cn(CN2CCCC2)nn1)=O CCC(CC)C(=O)NCC(CCOC)NC(=O)CCn1ccc(C)n1 C1(CNC(C=C(C)C(C)C)=O)CC(C(=O)N(C)Cc2cnc(C)o2)=NO1 C(CC(C)C)(C(=O)NC(C)C(=O)NCC(C)(C)C(N)=O)OC C1(NC(C2CCCC(C)(C)O2)=O)CN(C(c2ncc[nH]c2=O)=O)C2(CCCC2)C1 c1(N(C(c2cscn2)=O)CCC2CCCNC2)ncnc2cccc(F)c12 NC1CCC(CNC(=O)C(N2CCC2C(=O)NCCc2ccccc2)=O)CC1 c1(N2C(C)CC(CNC(c3n(CC)nnc3C)=O)C2)cc(C)nc(C(C)(C)C)n1 CC(=O)n1cc(Cn2cccc2CNc2nccc(C)c2F)c2cccnc12 n1(CCCC)nc(C(=O)NC2CC2CSc2ccccc2)c2ccccc2c1=O N1(C(CN2CCC(OC)C2)=O)CCOC(C)(CNC(c2ncc(C)cc2F)=O)C1 Cc1ccnc(C(C)NC(C23CC(CN2C(C24COCC2C4)=O)C3)=O)n1 C(C(C)(C)C#CC(=O)Nc1cccc(F)c1O)NC(CS(CC)=O)=O CC1(C)C(CNC(C23CCC(C2)C3)=O)CCN1C(c1cc(O)cc(F)c1)=O C(=O)(C(C)(C)CC(=O)N1CCOCC1CC(=O)NCCCCCCO)OC C1(C(N(CC(=O)NCC2C(C)(C)C2(F)F)CCC)=O)C2(CC2)C12CC2 Cc1ncnc(O)c1C(=O)NCC1CC(C)(C)CN1C(c1ccoc1)=O C1(C(=O)Nc2cc(C3(CC)CC3)no2)CC(=O)N(Cc2ccccc2)C1 N1(C(C2C(C(=O)OCC)CC2)=O)CC(C)(NC(=O)CC2COCC2O)C1 N1(C(c2c(C)occ2)=O)CCCC2(CCCCC2NC(=O)CC(C)C(F)(F)F)C1 C1(NC(=O)CC2CC(NC(c3ccc(F)c(Cl)c3)=O)C2)CCc2ccccc2C1 O=C(C1=C(Cl)CCCC1)NCC1(CNC(=O)C2CC2)CCCCC1 CCC(CC)CC(=O)NCCCOCCNC(=O)C(C)C(C)c1ccc(Cl)cc1 C(=O)(CC(F)(F)CC)N1C(CC)C(C(=O)NCC(O)CN(C)C)CC1 N1(C(=O)OC(C)(C)C)CC2CC1CCC2Oc1ncc(OC(C2CCCO2)=O)s1 CC(CCC(=O)NCCn1cnnc1O)NC(=O)C=Cc1cscn1 CC(CS(C)=O)C(=O)NC1CN(C(=O)CC#N)CC1c1cnn(C)c1 Cc1c[nH]cc([N+](=O)[O-])c1=NC(C)CCNC(c1cc2c(F)ccc(F)c2[nH]1)=O N1(C(CCCOCCOC)=O)CC=C(C(C)(C)C(=O)N2CC(OC)CC2CO)C1 CC12CCC(n3cc(CNC4CCC=CO4)nn3)(CO1)C2 C(CN=c1cc(Cl)nc(C(F)(F)F)[nH]1)(C1CCC1)NC(C(C)(O)C1CCC1)=O N1(C(C2CCN(C(C)=O)C2)=O)CC2CC(C1)C2NC(=O)C(C(C)C)n1cnnn1 c1(C(=O)NCCC(C(C)C)NC(=O)C(C)C(C)(F)F)ccc([N+](=O)[O-])c(Cl)c1 c1(OC(C)C(=O)NCC(C(C)(C)C)NC(c2cc(Cl)c[nH]2)=O)ccc(F)cc1 N1(C(c2scc(COC)c2)=O)CCC(NC(=O)CCCSC)C(F)(F)CC1 N1(C(CC2C(C)C2(F)F)=O)C2CCC1CC(CNC(c1nnc(S)n1C)=O)C2 C1(CC(=O)NCCn2cnc(-c3nn[nH]n3)n2)CN2CCN1CC2.C1C(=O)N1 C1(C(CCC)NC(=O)C(O)Cc2[nH]cnc2C)CCN(C(=O)C(=O)N(C)C)CC1 C1(CN(C)C)CCCN(C(=O)Nc2nccs2)C1.C12(CCC1)CN2 c1(-c2nc(NCC(=O)Nc3nnc(CCCC)s3)sc2)ccccc1F n1(C(C)C)cc(CNC(=O)CC2CC(NC(=O)C(=O)C3CCCC3)C2)cn1 C1(CNC(C(CCC)(C)O)=O)CN(C(=O)COC2CC(F)(F)C2)CCC12CCC2 C1(C(N2CCCC2CNc2ccccc2)=O)CC(NC(=O)CC(F)(F)F)CCO1 N1(C(C=Cc2ccc(C)s2)=O)CC2CCN(C(C3CC3c3ccnn3C)=O)CC12 N1(C(c2cc(C)n(CCO)n2)=O)CCN(C(c2ccsc2)=O)CC1CS(C)(=O)=O C1(F)(C(=O)NCc2cnc(CNC(=O)OC(C)(C)C)[nH]2)CCCOC1 Cc1nn(C)cc1CC(=O)NCC1C2CN(C(C3CN(C(N)=O)C3)=O)CC12 N1(C(CC2CC(=C)C2)=O)CC(C)CN(C(c2ccc(C)nc2OC)=O)CC1C CCCCC(C)C(=O)N1CCOCC(CNC(=O)CCc2ccc(OC)cc2)C1 N1(C(C2CCNCC2OC(c2onc(C(=O)NC)n2)=O)=O)CCC(CO)CC1 CC1CN(C(C2(Sc3ccccc3F)CCC2)=O)CCCN1C(=O)CNC1CC1 Cn1cc(NC(C23CC2CN(C(c2cccc4c2OCO4)=O)C3)=O)c(O)nc1=O C(=O)(C(CCC(C)C)NC(c1cc(C)[nH]n1)=O)NCc1cccc(CC)c1 C1(CNC(c2n(CC)nnc2C)=O)CCN(C(=O)COCCF)CCC1(F)F N1(C(C2(CC#C)CCCC2)=O)CCCC(CNC(c2cc(C(F)(F)F)c[nH]2)=O)C1 C1(C)(CN(C2(C3CCCO3)CCC2)C(C)=O)COCCN(C(C2CCOCC2)=O)C1 C1(CNC(C=CSC)=O)CCCC2(CN(C(c3n[nH]c4c(C)cccc34)=O)C2)O1 N1(Cc2nc(C)c(F)cc2)CCC2(CC1)CC2(C)C(=O)NCC1CCCCO1 c1(C(N2CC(OC)C(NC(C34CCC(CC3F)C4)=O)C2)=O)cc(C)c(N)cn1 CC1(CNC(c2cccc(C3CC3)c2)=O)CCCN1C(=O)Cc1nc[nH]n1 c1(C(N2CC(O)CC2Cn2cc(CN3CCNC3=O)nn2)=O)ccc(Br)cc1I c1(C(=O)NC(C(C)NC(c2nc(C)n(C)n2)=O)C)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(C#CC(=O)O)=O)CCCCC(NC(c2c(O)cccc2Cl)=O)C1 c1(C(=O)NC2CC(CC)NC2)cc(-c2cccc(F)c2)n(C)n1 CCC(C)(CC)C(=O)N1CCC(C2CCCCN2C(C2C3CCCC23)=O)C1 N1(C(C(Cc2ccc(OC(C)C)cc2)NC(CSC)=O)=O)CCCC2OCCC12 C1(C)(C(N(c2ccc(F)nc2)C)=O)C=CCN1C(c1ccnc(O)c1)=O c1(CNC(=O)C=CC2CC2)ccc2c(c1)CCC2NC(=O)C1CCc2c[nH]nc21 c1(N(COC)C2CC2)ccccc1-c1ncsc1-c1nc(C2CC2)nn1C C(CCCCCN(C(=O)CC1CCOC1C)C)NC(C(=C(C)C1CC1)F)=O N1(C(CCC(C)OC)=O)CCC(C)(C)C(C(=O)NC(C)(C)CCF)C1 c1(C(=O)NC2CC(NC(CC(c3ccc(C#N)cc3)C)=O)C2)ncnc(O)c1F c1(C(=O)NC)cccc(C(N2CC=CC(NC(=O)C3=COCC3)C2)=O)c1 C1(C(=O)NC2C(NC(C=C3CCC(C)CC3)=O)COCC2)CCC2(CC1)CC2 N1(C(C(CCC)C)=O)CCC(CNC(C2CC2C(F)(F)F)=O)C12CCC2 N1(C(C2N(C(=O)N(CC3(C)CCN(C)C3)C3CC3)CC2)=O)CCC2CC1C(=O)N2C CC(C)C(F)C(=O)N1CCOCC1CC(=O)NCCCC(C)(F)F Cc1cc(Br)cc2cc(CN3CCC(C(=O)O)CC3C)[nH]c12 C1(C(=O)NCCOC2CN(C(=O)CC3CCCN3C)C2)(CC)CC2(CCC2)C1 Cc1ncn(C)c(=O)c1C(=O)NCCC(C)CCNC(c1cc(O)nn1C)=O N1(C(C2CCOCC2)=O)CCC(O)(C(=O)NCC2CCCNC2)C1 C1(CN(C(COCC(=C)C)=O)C)CCCN(C(=O)COC2CCN(C)CC2)C1 N1(C(Cc2cnc(C)s2)=O)CC2CCN(C(C3CCCS(=O)(=O)N3)=O)CC2C1 c1(-n2ncc(C(N3CC(CC(C)NC(C=CSC)=O)C3)=O)c2)cccc(F)c1 C1(CNC(CCC(=O)OC)=O)CCC(C)N(C(c2ccn(CC(C)C)n2)=O)C1 n1(CC(=O)N(C2CCN(C(=O)Cc3c[nH]nc3C)C2)CCC)cc(F)ccc1=O N1(CCNC(C(c2c(CC)n(Cc3ccccc3)nc2)OC)=O)CCN(C)C(=O)C1 C1(C(N2CCN(S(C)(=O)=O)CC2)=O)CN(C(=O)Nc2ccncc2)CC(F)(F)C1 c1(OC)ccc(NC(CCC2N(C(c3ccc(Cl)cc3)=O)CCC2)=O)cc1OC CC(C)CC(Cc1cccs1)C(=O)NCC(C)N(C(=O)C(C)Cn1cccn1)C c1(NC(C2C3CN(S(=O)(=O)Cc4cccc(F)c4)CC23)=O)ccnc(CO)c1 C12(CNC(C3C(OC)CC3)=O)CC(CO1)N(C(=O)CC(C)c1ccccc1)C2 C1(NC(c2cnn(C)c2N)=O)CC2(C1)CN(C(C1CCC1C(C)(C)C)=O)C2 C1(O)(CC(=O)N(CC(CC)NC(=O)C=CCN(CC)CC)C)CCCN(C)C1 CCCCC(C(=O)N(C1CCCC(O)C1)C)NC(=O)COCCSC C1(C(=O)NCC(C2CCC2)NC(C=Cc2cn(C)nc2)=O)CN(S(N)(=O)=O)C1 C1(CC(=O)NCc2cncc(CO)c2)C2CN(C(C3C(C(N)=O)COC3)=O)CC12 C(=O)(CC(C)(C)CC)N1CC(CNC(c2ccc(CC)nc2)=O)C1 N1(C(C(C)SC)=O)CC(C)CCC1CNC(C1(C2CC2)CC1)=O CCCC(C)(C)C(=O)NCC1CN(C(C2C3(CCC3)C2C(F)(F)F)=O)CC1C C1(C(=O)NC2CCC2CF)CCCC1CNC(=O)C(F)(F)c1ccsc1 c1(C(=O)NCC(C2(O)CCN(C(=O)COC3CCCC3)C2)C)ccc(OC)cc1 C(C)(CNC(C1CCOC1C(C)C)=O)(CC(C)C)NC(c1c(CC)csc1)=O C(CCNC(c1cccc(=O)o1)=O)(C(=O)NCC1COCCO1)OC c1(C(=O)NCC(CNC(c2ccc(CC)s2)=O)F)cc(C)nc2c1CCCC2 C=CCCC(C)(C)C(=O)NCc1nc(C(=O)NC(CN2CCCC2)CC)co1 C(=O)(C(F)C(=O)NCCC1CCCCN1C(c1c[nH]nc1CC)=O)OCC C(C(=O)N1CCC(CC(C)NC(=O)CC2CCOC2)CC1)(C(C)C)OCC c1(C(C)OCC(CC)NC(=O)NC2CC2)cnn(-c2ccc(F)cc2)c1C c1(C(N2CCN(C(c3cc(C)c(C)[nH]3)=O)C(C)C2)=O)nn2cccnc2c1Cl c1(C(C(=O)N(C(CNC(C2CC23CC3)=O)C2CC2)C)C)ccc(Cl)c(Cl)c1 c1(N2CCCC(CCNC(c3cc(F)cnc3O)=O)CC2)ncnc2c1COC2 N(C1CCCn2nccc21)C(C(CC=C)CNC(=O)C(C)N(C)C(C)=O)=O N1(C(=O)N(C2CCN(C(C(c3ccccc3)N(C)C)=O)CC2)CO)CCCS1(=O)=O c1(C(=O)NCC(CC)(CC)NC(=O)CC2CC2(Cl)Cl)ccc(NC)c(F)c1 CC(C(=O)NC(Cn1cncn1)C(=O)NCC(F)C1CCC1)S(C)(=O)=O Cc1c(C(=O)NCC2CC2NC(=O)CCC2CC2(F)F)ccc(Br)c1F c1(CCNC(C(CSCC)NC(c2cnccn2)=O)=O)ccc(F)cc1 CCCCC(C(=O)NCC1(CNC(=O)C(n2cc(C)cn2)C)CCC1)C(C)C c1(C(N2CC(C=C)C(NC(=O)C(C)(C)C(F)F)C2)=O)ccc(S(N)(=O)=O)c(C)c1 c1(NC(C2C(NCc3c(OC)ccc(Br)c3)C2)=O)ccc2c(c1)COC2=O c1(C(=O)OC)ccc(C=CC(=O)NC2(CNC(c3cn(CCO)nn3)=O)CC2)o1.OC c1(N(C)CCC2CCCN2C)nc2cccnc2c(=NC2CC(=O)N(C)C2)[nH]1 c1(C(N2CC(COC)(NC(=O)C3=CC(O)C3)C2)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(=O)NC2(CCCN3CCCC3)OCCO2)CCN(C(c2ccsc2)=O)CC1 CC1(C)CC(N=c2nc(N3CC(C)(C)OC(CO)C3)c3cc(F)cc(F)c3[nH]2)CCO1 c1(C(=O)NC(C)C(=O)NCC(C)(Br)Br)ccccc1Cl N1(C(CC2(COC)CC2)=O)CCC2(CC1)CN(C(c1sc(COC)nc1C)=O)C2 C(CC(=O)NC(C)CCN(C)C)(C(F)(F)F)NC(c1cc(OC)ns1)=O c1(CNC(c2cccc(SC)n2)=O)ccc(F)c(C)c1.C12(CC)CC(C1)NC2=O c1(N2C(CN(C3CCCC4CC34)C(C)=O)CCC2)ncc([N+](=O)[O-])c(C)n1 CN1CCC(C(=O)NC2(CC(=O)NC3(C)CC3)CCC2)C1 C1(C(=O)NCCCN(C)C(c2ccc(N3CCCC3)cc2)=O)CC(C2CC2)=NO1 c1(C(=O)OCC)ccc(S(=O)(=O)N(CC)Cc2ccc(F)c(F)c2)cc1 C(CCC)(CCCNC(=O)Cc1c[nH]nc1C(F)(F)F)NC(CCC#CC)=O C12(NC(CC3(O)CCCN(C)C3)=O)CCCCC1CN(C(=O)CC(F)F)C2 C1(C)(CCNC(C2CCC(OC)C2)=O)CCN(C(=O)CCOC2CC2)CC1 N1(C(C(C)=C2CCC2)=O)CC2(C1)CN(C(=O)CC1CSC1)CC2CO N1(Cc2cc(C)n(CC)c2C)C(=O)CNC(=O)C1C N1(C(C2C(C#C)C2(C)C)=O)CCN(C(=O)CNC=O)C(c2ccc(OC)cc2)C1 c1(C(=O)NC2CC3CC2CN(C(c2cncnc2)=O)C3)cnn2cccc(Cl)c12 C(C)(CCC(=O)NCCC(=O)NC(C)(C)C)SC.c12ccc(nc1)[nH]c2=O N1(C(CCN(C(=O)C(C2CC2)OC)CC)=O)CCC(O)CC1 C1(CCNC(c2ccsn2)=O)COCCN1C(C1CCOC1C1CC1)=O C(=O)(C(C)(C)C(C)(C)C)N(CC(C)NC(c1cc(F)cnc1O)=O)C Cc1cc(C(=O)NCCCCC(C)NC(c2cscc2F)=O)oc1C Cc1cc(CN2CCC(O)C(F)C2)cc(C)n1.N12CCCC1CNCC2=O CN(C)S(=N)(=O)c1ccccc1C(N1CCC2(CC1)OCCCC2O)=O C1(NC(CCC(C)NC(C(COC)(C)OC)=O)=O)CC2(C1)CC21CC1 c1(C(N2C3CN(C(=O)NCCCl)CC32)=O)cnc(O)cc1O c1(N2C3CN(C(C)=O)CC32)ccc(=NCc2cccc([N+](=O)[O-])c2)[nH]c1 c1(OC2CCN(C(C3C(C)C3)=O)C(=O)C2)cccc2cnccc12 c1(OC)ccccc1OCCC(=O)NC1(CNC(=O)CCNC)CC1.C1(CN)CC1 C(CCN=c1nc(N2CCS(=O)(=O)C(CSCC)C2)c2c([nH]1)CCCCCC2)SC COn1cnc(C)c1C(=O)NC1CN(C(=O)CCOc2cccc(Cl)c2)CC1F N1(C(C2C(=C)C2)=O)CCC2(CCOCC2)C(NC(=O)CC2CCN(CC)CC2)C1 C1(C(N2C(CC(=O)N(C)Cc3ncc[nH]3)CC(F)C2)=O)CCCC2(CC2)C1 c1(CC(=O)N(CCN(c2ccccc2)C)C2CC2)ccc2nc(Cl)sc2c1 C(CCN=C(NCCCl)NC1(C)CN(C(=O)Oc2cccnc2)C1)NC.C(C)(C)(C)O C1(NC(C2C(C)(C)C2)=O)CC2(NC(=O)C=C3CCSCC3)COC1C2 CC1CN(C(=O)CC2CCOC2)CC1CNC(c1ccc(-c2ccncc2)o1)=O c1(C(N2CC(NC(C3CN(C)CC(C)O3)=O)C2)=O)c2c(cc3c1CCC3)CCC2 c1(C(N2CCC(C3CCCCO3)C2)=O)ccc(Cn2cccn2)cc1 C1(OC)(CNC(=O)C=CC2CCCC2)CCN(C(=O)CC2CCC(C)C2)CC1 N1(C(C2N(C(C=Cc3ccc(C)o3)=O)CCSC2)=O)CCC(C)(F)CC1 Cc1cc(C(=O)NC2CCN(C(=O)CN3CCCC3)CC2)n(-c2ccccn2)n1 C1(NC(c2ccn(C)c2)=O)CC2CC(NC(=O)CCCC(=O)N(C)C)CC12 C(=O)(C(O)C1=CCCCC1)N1CC(O)(C(C)N(C(C(=O)NC(C)(C)C)=O)CC)C1 c1(C(CC(=O)NCCN(C(=O)Cc2ccns2)C)C)c[nH]c2ccccc12 N1(C(c2cc(C)sn2)=O)CCC(C(C)(C)CNC(C2(O)CCCC2)=O)CC1 Cc1cc(O)ncc1C(N1C2CC1CN(C(=O)Cn1cnc([N+](=O)[O-])c1)C2)=O C12CC3(CC(C3)NC1=O)C2.c1(CN2CCC(F)(C(=O)OC)C2)ccc(F)c(O)c1 c1(NC(N)=O)ccccc1C(=O)NC1CC(NC(c2ccncc2)=O)C1 CCC(CC(=O)NC1CN(C(c2ns[nH]c2=O)=O)CC1N=[N+]=[N-])CC(C)C C1(NC(=O)C(c2ccccc2)O)CCN(C(C2CC=CCO2)=O)CC1F c1(CC(=O)NC2CCN(C(=O)Cc3cscn3)CC2F)cc(Cl)c2c(c1)OCO2 N1(C(C(C(C)C)OCC)=O)CC2(CCNC(=O)Cn3cccc3)CCC1CC2 Cc1cn(C)nc1C(=O)NCC1CC1NC(=O)C(C)CN(C)C C1(S(N)(=O)=O)(C(=O)NCC2(CN(C)CCOc3ccccc3F)CC2)CCC1 C1(NC(C2C(CC)CN(C(=O)C(C(C)C)SC)C2)=O)CC2(C1)CC(O)C2 c1(C(N2CC(O)CC(NC(COCCC#C)=O)C2)=O)cnc2ccccc2n1 Cn1c([N+](=O)[O-])cnc1C(=O)NCC1CC(NC(C2CC(CC3CC3)C2)=O)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CCCSC1)NCc1nc(CC)on1 CC(C)(C)C(CC(F)(F)F)C(=O)OCCC1CCCC12CCC2 c1(C(N(CCNC(C(C)OCC#C)=O)CC2CC2)=O)cncc2nc(C)[nH]c12 N1(C(c2cnn(C(C)C)c2Cl)=O)CCCC(NC(=O)CN2CCC(C)(O)C2)C1C Fc1ccc(CN2CCN(Cc3ccsc3)CC2)cc1Cl N1(C(c2cnc(C)o2)=O)CCC(NC(c2onc(Br)c2C)=O)C(O)C1 N1(C(c2ccn(CC)n2)=O)CC(OC)CC(NC(c2cnn(CC(C)C)c2)=O)C1 c1(CS(C)(=O)=O)ccc(NC(=O)NC2(Cc3ncco3)CC2)cc1 C(=O)(CC(F)(F)F)NC(C)C(=O)N(C(C)CCNC(C1CC1C(C)O)=O)C C=C=CCC(=O)N(C1(CNC(=O)CSc2ccccc2)CC1)C C#CCC(CC#C)C(=O)NCC1CC(CNC(c2cc(N)cc(F)c2)=O)C1 c1(CCNCCCC(c2nnnn2C(C)C)OC)cccc(F)c1 c1(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)(F)F)C)ccc(C(C)(F)F)cn1 CN1Cc2cc(OC3C(C#N)C34CCC4)ccc2C1=O CC(CCNC(=O)C(C)N(C)C)CCNC(=O)CC(C)(F)F c1(C(=O)NCc2cn(-c3ccc(C(=O)O)cc3)nn2)cccc2c1CCS2(=O)=O N1(C(C2CC(=C)CN2C(C2CC(F)C(C#N)C2)=O)=O)CCC2(CCCO2)CC1 n1(C(C(=O)NC(CNC(C=C(CC)C2CC2)=O)CC)C)ccnc1C CC(CS(C)(=O)=O)C(=O)N(C1CCN(C(=O)CCCCCF)C1)CCO C1(CC(=O)N(CCNC(c2sccc2OC)=O)C(C2CCC2)C)CCCC1CC N1(C(C(C)OCC#C)=O)CCN(C(c2cnc(C)[nH]c2=N)=O)C2CCCC12 Nc1ccc(C(=O)NCC2CCCN2C(c2coc(C(F)(F)F)n2)=O)nc1N c1(NC2CCC(C(=O)NC(=O)NCC3OCCN(C)C3)OC2)ccc([N+](=O)[O-])cc1 C(=O)(C1=CCCOC1)N1CC(C)C(CNC(=O)CCc2cccc(Cl)c2)C1 C=CCCC(C(=O)NCC12CCC(CC1)C2)NC(C1OCC2(CCC2)C1)=O CC(C)CC(C)(C)C(=O)NC(C)C(C)C(=O)NC1(C)CCCC1 C(=O)(CCC(=O)N1CCOCC1)NCC=CCNC(c1ccc(C(C)(C)C)s1)=O CS(=O)(=O)CCC(=O)N1CC2CCC2(CNC(C2(F)CCC=CCC2)=O)C1 N1(C(C)=O)CSCC1C(=O)NCC1(NC(=O)Cc2ncc(C)s2)CC1 N1(C(c2ccnc(CC(C)C)n2)=O)CC(NC(=O)Cc2csc(S)n2)C(C)(C)C1 CC1CC(CNC(=O)Cc2nc[nH]n2)CN1C(c1ccoc1Cl)=O C1(F)(CNC(C2C3CCCC23)=O)CCN(C(c2cnn3ccsc23)=O)CC1 C1(CC#C)(C(=O)NC(C2CSC2)C)CCN(C(c2cnc(C)nc2)=O)C1 N1(C(c2ncc(C)c(Br)c2)C(=O)NCCC#N)CCc2cc(F)c(F)cc2C1C c1(OC)ncc(Cl)c(=NC2CCC(NC(c3cc(C)ccn3)=O)CC2)[nH]1 N1(C(COCc2cc(C)on2)=O)CCCC(CCNC(=O)C(C)C(C)C)C1 CCC(CC)(CC)C(=O)NCC(C(=O)NC(c1csnn1)C)N(C)C C1(C(N(CCCO)C)=O)CCCN1C(=O)C=CC(F)F.C(=O)N Cc1cccc(C(F)C(=O)NCC(C)CN(C)C(c2c(C)nsc2C)=O)c1 CCC(F)(C(=O)OC)C(=O)NCC1CCN1C(c1cc2cccnn2n1)=O c1(CC(=O)Nc2c[nH]nc2C(=O)Nc2nc(Cl)ccc2Br)c(F)cccc1F CC(C)CC(C)CC(=O)NC(C)(C)CN1CCN(C(c2cnc(Cl)s2)=O)CC1 O=[N+]([O-])c1c(CNC2COCC2N2CCOCC2)ccc(O)c1O C1(NC(C2(COC)CC2)=O)CCOC2(CCN(C(=O)CNc3nccs3)CC2)C1 C1(NC(c2cncnc2C2CC2)=O)C2CN(C(c3csc(C(F)(F)F)n3)=O)CC12 c1(N2CCC(COC)C2)cc(CNN2CCC(O)CC2)ncn1 Cc1ncc2n1CCN(C(=O)CC=CCNC(C1CC(=O)CCO1)=O)C2 C1(C(N2CCCC(NC(=O)CCc3ncc[nH]3)CC2)=O)CCc2nc(O)[nH]c2C1 CCCC(F)C(=O)N1CCCC1CNC(C1(OCC)CCCCC1)=O N1(C(C(C=C)(C)CC)=O)CCC2C(C1)NC(=O)CN2C(=O)CCCCOC N1(C(c2c(C)csc2)=O)CCC(CCNC(=O)C2=CC(O)CCC2)C(F)(F)C1 CC(C)(CC(=O)N1CC(NC(C2(O)CCCC2)=O)CC12CCOC2)CC(F)F N1(C(CC(C=C)(C)O)=O)CC(CNC(c2ccoc2C2CC2)=O)OC2(CCC2)C1 c1(N2CC(CNC(C(CC)C)=O)C2)ncnc2ccc(OC(=O)C(C)C)cc12 C1(NC(c2c(OC)nccc2)=O)CC2CCC1N2C(c1ccco1)=O N1(C(CNC(C)=O)=O)CC2CC(NC(c3cc(C(F)(F)F)ccc3Cl)=O)C1C2 C(CCN=c1ccnc(NCCSCCCN2CCOCC2)[nH]1)OCC C1(CNC(CCN(CC)CC)=O)CCC(C)(C)CN1C(=O)Cn1cccnc1=O Cc1cc(Br)cc(F)c1NC(C1CCCN(C(c2nn[nH]c2C(F)(F)F)=O)C1)=O c1(SCC(=O)N(C2CN(C(=O)CC3CCCCO3)CC2F)C)cccc(F)c1 N1(C(C(C2CC2)OCC)=O)CCC2(C1)CN(C(=O)C#CC1(C)COC1)CCO2 C1(C(N(C(C(=O)N(CC)CC)C)CC)=O)CC(C)CC(=O)N1 Cc1nc2ccccc2c(C)c1CC(=O)NC12CC1CN(C(=O)C=CS(C)=O)C2 c1(C(=O)NCC(CC(C)C)(C)NC(=O)COCCCF)occ2c1CCOC2 CC1CC(C(=O)NCC2=CCCN(C(=O)COc3ccccc3)C2)CC(C)C1 C1(O)(C(=O)NCC2C(CNC(c3c[nH]c(=N)s3)=O)C2)CCSCC1 C1(C(=O)NCC2N(C(C3OCCN(C)C3=O)=O)CC2)CCC(C2CCCO2)O1 c1(CC)conc1CC(=O)NC1(CNC(=O)C(C)Cc2cnco2)CCOC1 c1(C(=O)OC)cc(=NC(=O)c2n[nH]cc2NC(=O)Cc2cnn(C)c2)[nH][nH]1 N1(C(c2ncc(C)s2)=O)CCN(C(c2c(C)nc(C(C)C)nc2O)=O)CC1C#N CN1CCC(O)(C(=O)NCC2(F)CCN(C(=O)CNC=O)C2)C1 CC(C)(C)C(CO)C(=O)NC1CCCC1NC(c1c(Br)cnn1C1CC1)=O c1(C(=O)OC)c(CCC(=O)NC2CCCOC2C(C)(C)C)c[nH]c1C C1(CC)CCN(C(=O)OC(C)(C)C)C1C.C12(CSC1)NC2 CC12CC(CNC(c3ncoc3C)c3nnnn3C3CCC3)(CO1)C2.C1CC1 c1(OC)cc(C(=O)NCC2CCCC2NC(c2cc(C)ns2)=O)sn1 C1(NC(C2N(C(CCC)=O)CCC2)=O)CC(F)CN(C(C2CC(C)(CC)C2)=O)C1 CC1(C)OCCC1CC(=O)NC1CCCC1NC(c1cnn(C2CCCC2)c1)=O C=C1COCC1NC(c1nnnn1C)(C1CN(c2ccccn2)C1)C c1(C(N2CC(O)(C(=O)NCCC3CCC(C)O3)C2)=O)ncncc1N C(=O)(CCC1=NNC(=O)CC1)N1CC(NC(C(CC)CC)=O)C2C1C2 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(CNC(=O)CC2CCC2)C(O)C1 CCC(CC)CCC(=O)N(C)CCC1CCN(C(C2(CC)CC2(F)F)=O)CC1 N1(C(=O)OC(C)(C)C)CCCC1C=CC(N1CCOCC1C(F)F)=O c1(OC)cc(OC)c(C(N2CCC(NC(C3CCCO3)=O)C(OC)C2)=O)c(N)c1 C1(C(=O)NCCCN(C(=O)Cc2cnn(C(F)F)c2)C)CN2CCCCC2CO1 c1(C(=O)NC2C(CNC(c3c(C)n(C)nc3)=O)C2)cc2c(C)c(Cl)ccc2[nH]1 c1(C(N(CCCC(=O)OC)C2CC2)=O)cccc(OCC(N)=O)c1 C1(C(=O)NC(CC(C)NC(C(CC)=CCCC)=O)C)CCCOC1C c1(C(N2C(CNC(=O)CC3(C)CC3)(CSC)CCC2)=O)ccc(OC)c(Cl)c1F c1(COC)nc(=N)[nH]cc1C(=O)NC1CC1NC(=O)CCc1nccs1 C(C)(CC(=O)N(NC(=O)OC(C)(C)C)C(C)C)c1c(C)cccc1C c1(OC(C2(CN(CCC)Cc3c(C)noc3N)CC2)=O)ccc(Br)cc1F Cc1cnc(C(=O)NCCC(C)NC(=O)C(C)OCCN(C)C)cc1Cl Cc1ccc(C(CN2CCCCC2)Nc2ccc(-n3cnnn3)cc2)cc1 Cc1cc(C(N2CCOC(C(C)NC(C34CC(CO3)C4)=O)C2)=O)ccn1 O(S(=O)(=O)c1ccccc1F)c1cccc(NC(c2cccc3cncn23)=O)c1 c1(OC)cc(CNc2cccnc2C(N2CC(F)(F)C(F)(F)C2)=O)cc(O)c1O C1(NC(C2(CCCC)CC2)=O)CCCC2CN(C(c3sccc3C(C)=O)=O)CC12 N12CCC(CCOC)(CC1)N(C1CCC1)CC2=O.CCC(C)C(CO)NC(=O)CO c1(C(=O)NC2(CNC(C3CC(SCCO)C3)=O)CCC2)ccc(Br)nc1 C(=O)(C(C)(C)C1CCCCC1)N(CCN(C(=O)CSC1CCCO1)C)C c1(C(N(CC(C)NC(=O)C(C)(CC)OC)CC)=O)cc2c(s1)CCCCC2 c1(C(=O)NC2C(NC(C(CCSCC)NC(N)=O)=O)C2)ccc(S(N)(=O)=O)o1 CC1(C)CN(C(=O)C(N2CC3CC(F)(C3)C2)=O)c2ccccc2S1=O C1(NC(CCN(CCC)C)=O)CC2(CCCN(C(=O)C(C)=C3CCC3)C2)C1 c1(C(=O)NC2CC(C)(NC(C(CCCCC)O)=O)C2)cccc2nc(C)[nH]c12 c1(OC)ccc(CCC(=O)N(C)Cc2ccc(Cl)cc2Br)cc1F C=CCCCCC(=O)N1C2CCC1C(CNC(=O)CS(=O)(=O)N1CCCCC1)C2 c1(C(N2CC=CC(NC(CC(=O)N(C)C)=O)C2)=O)c(C(F)(F)F)cccc1Cl CC1(C)CCCN(C(C2(C#N)CCC2)=O)C1CNC(c1cccnc1S)=O N(C(=NCCCNS(=O)(=O)C1CC1)NC1CC1)C(c1c(F)cccc1Br)C c1(C(=O)NC(CNC(CCC)=O)CC(C)C)cnn2c(=N)[nH]cnc12 C1(CC)C(NC(=O)COC2CCOC2)CCCN1C(=O)CCCCOC CC1(CNC(C2(CC(F)(F)F)CC2)=O)CCN(C(=O)C=CC2CCC2)C1 CC1CN(C(=O)C(=O)NCC(F)F)CC(C(=O)NCc2cc(O)ns2)O1 Cc1ccc(C=CC(=O)NC2(C3CCCCN3C(C3CCC3(C)C)=O)CC2)o1 Cc1cc(O)c(F)cc1NC(=O)C(C1(C)CC1)NC(c1ccc2cc[nH]c2c1)=O C(=O)(C(C#N)C(C)C)C1CC1.C(=O)(C(=O)NCCCNC(=O)CCOCCS)OCC N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(C)(C)C(CNC(C2CCN(C)CC2)=O)C1 c1(C(N2C(CCC(=O)N(CC(N)=O)C)CCC2)=O)ccnc(Br)c1F CCC(CC)C(=O)N1CC(COC)(NC(C2C3CC4C(C3)C24)=O)C1 N#Cc1cc(C(=O)NC2CC3(C2)CN(C(c2cc4c(s2)CCC4)=O)C3)ccc1F N1(C(c2nccn2CC2CCCC2)=O)CCC(n2cc(CC(CO)C3CC3)nn2)C1 Cc1cc(Br)c(NC(C2CN(C(c3ccc(O)c(F)c3F)=O)CCN2)=O)nc1C CN1CCOC(CN2CCC(C)(NC(c3ccsn3)=O)C2)C1 c1(C(=O)NCC(C2CC2)NC(C=Cc2c(C)cccc2)=O)ncc(C#N)cc1Cl C(=O)(CC1OCc2ccccc21)NCC(CC)Nc1cc(C(C)(C)C)[nH]n1 N1(C(=O)Cc2cn[nH]c2)CCC2(CCCC2NC(=O)C(O)(C2CC2)C2CC2)CC1 CC(C)C(C)(C)C(=O)NCCCN(C(=O)C(=O)NCC1CC1)C N1(C(c2ccnc(C)c2N)=O)CCCN(C(=O)CCc2nc[nH]n2)C(C)C1 c1(C(=O)NCCCC(CCC)NC(=O)CCSC)cnn2ccc(OC)cc12 CCC(C)CCCC(=O)NCCCN(C(=O)C(C(C)C)N(C)C)CC c1(C(=O)NCC(CNC(C2N(CC)CCCC2)=O)(C)OC)ccc(C#N)c(C)c1 c1(CC(C)C)ccccc1C(=O)OC(C12CCC(CC1)C2)C c1(N2CC3(CCN(C(C4C(C)(C)CCC4)=O)C3)C2)ccc2c(n1)CCC2=O C#Cc1ccc(F)cc1C(=O)NC1(C)CC(NC(=O)CCc2cccn2C)C1 c1(N2CCOC(C)C2CO)nc2ccc(Cl)c(Cl)c2s1 c1(CC(C)(CN)NC(=O)CNC=O)ccc(C(F)(F)F)cc1.CCC(O)C=O c1(C(=O)NC(CO)C2CCC2)ccc(F)c(O)c1 N1(CC(=O)NCC(CNC(C2CC(C)(F)C2)=O)O)CCN(C2CC2)C1=O c1(N2CCC(NC(=O)C(F)C3CCC3)(CF)C2)ccncc1[N+](=O)[O-] Cc1nn(CC(F)F)cc1C(=O)NCC1(O)CCN(C(C2(Cl)CC23CCC3)=O)C1 CCCC(O)C(CO)NC(=O)C(F)C(C)CNC(C1CN(C)CCN1C)=O CC1(C)CC(O)(C(N2CC(CNC(c3ccncn3)=O)C2)=O)C1 c1(C(c2ccccc2)C(=O)NCC2C(C)C2(F)F)c(F)cccc1Cl CC(C)CC(C(=O)NCCCCCCO)ONC(=O)Cc1ccccc1O N1(CC)CCOC(C(=O)NCC2C3CN(C(=O)CC4CC5CC4C5)CC23)C1 c1(OC)ccc(Br)c(CC(=O)NC2CCCC2NC(C2CCOC2)=O)c1 C1(C=C)(C(=O)NC(CC=C)CNC(c2nc(C)sc2C)=O)CCOCC1 c1(OC)ccc(CO)cc1C(=O)NC(C1CCN(C(=O)Cc2cccnc2)C1)C C1(O)(CCNC(C(C)N(C(C)=O)C)=O)CCCN(C(C2(CO)CCCC2)=O)C1 C12(C(N3C(CNC(C4N(CCC)CCC4)=O)CC3)=O)CC3CC(C1)CC(O)(C3)C2 CC1CC(C(=O)NC2(C)CC(C(=O)NCCc3cccnc3F)C2)CCS1 N1(C(Cn2cc(C)c(O)nc2=O)=O)CC2CN(C(=O)CC3CC34CC4)CCC12 c1(C(=O)NC2C(CCC)CN(C(c3cc(CC)oc3C)=O)C2)ccc(O)c(F)c1 c1(NC(C2CCCCCN2C(C2CC=CCO2)=O)=O)cccc2[nH]ccc12 C1(NC(c2nc(CC)oc2C)=O)CN(C(=O)CC2CCCCCO2)CC12CC2 N1(C(CCCCOC)=O)CCN(C(=O)C(=O)C2CC2)CC1CCO C1(CCN(C(C=CSC)=O)C)CCN(C(=O)C(Cc2ccsc2)NC=O)CC1 C1(NC(c2cc(Cl)ns2)=O)CCCN(C(c2csc(O)n2)=O)CC1 c1(C(=O)NC(C=CC(=O)NCC2(SC)CCC2)C)cc2ccccc2[nH]1 N1(C(C2CC(C)OCC2)=O)CCNC(=O)C1(C)C CCC(C(O)C(F)F)NC1(C(=O)O)CC2CCC1C2 C=CCC(C(=O)N1CCC(CCNC(c2coc(Br)n2)=O)C1)c1ccccc1 C1(C(=O)NCC2(C(N3CCCC(N(C)C)C3)=O)CC3(CC3)C2)CC(=O)NC1(C)C N1(C(C(CC#C)O)=O)CC2CC(C(=O)NC(C(N)=O)C(N)=O)(C2)C1 O(C=C(C#N)C(=O)N(C1CCN(C(=O)C(c2cccnc2)OC)C1)C)CC C#CC1CCCC(CNC(=O)C(C2(O)CN(C(c3ccc(F)cc3C)=O)C2)F)C1 C(=O)(C(F)CC(C)(C)C)NC1CC=C(C(=O)NCc2nn(C)c(=O)o2)C1 Cc1ccn2cnc(C(=O)NC(C)C(C)NC(c3cncnc3C3CC3)=O)c2c1 C(=O)(CCCCCNC(c1cc(CO)n(C)n1)=O)NC(CC(C)C)CN(C)C CC(C)CCC(C(=O)NCC(F)C(C)(C)O)NC(=O)C(O)Cn1cncn1 C1(C(=O)NC(C(=O)NC(CCC=C)C)CCOCC)CC2(C1)CC(C)C2 c1(C(=O)NC2CC(CCNC(CC(C=C)(C)C)=O)C2)c[nH]c2cc(Cl)ccc12 C(=O)(CCS(C)(=O)=O)NCCOCCNC(c1nc(SC)sc1)=O C1(c2nc(C(C3CC3)OC)nn2-c2ccnc(Br)c2)CC(C)OC(C)C1 C1(C(=O)NCc2cccc(OC)c2O)CC2(CO1)CN(C(=O)COC(C)=O)C2 CC1(C)C2CN(C(C3CN(Cc4cccc(C(C)(C)C)c4)CCS3)=O)CC12 Cc1cnc(C(=O)N(C2CCN(C(=O)COc3cccnc3Cl)C2)C)cn1 c1(C(N2C(CCNC(c3n(C)nnc3)=O)CCCC2)=O)ccc2c(c1)NCC2 c1(N2CCC(C)C(NC(C3CCCC(F)(F)C3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] C1(C(=O)NCCC2CC(F)(F)CN2C(=O)COC2CC2)COCCC1(F)F Cn1ncc2c1CN(C(=O)CC1CCNC(C(F)(F)F)C1)CC2 N1(C(Cn2nc(C)oc2=O)=O)CC2CCN(C(=O)C(C)(C)c3cscn3)CC12 C(C(C)(C)CC(=O)NC(CO)CC(C)(C)C)NC(c1cn(C(C)C)nn1)=O N1(C(c2n(C)nc(O)c2)=O)CC2(C)CN(C(=O)Cc3csnn3)CC2(C)C1 C1(C(=O)NC(C(OCC)OCC)C)CCCC12CCOCC2 Cc1nn2c(C(=O)NCC(C)(C)CNC(c3ccc(C)nc3C)=O)c(C)nc2s1 CCC(CNC(=O)C(CC1CCC1)NC(c1c[n+]([O-])c(C)cn1)=O)C(C)(F)F N1(c2c(OC)cc(F)cc2)CC(=O)Nc2ccccc2C1c1cccc(Cl)c1Cl C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCN(C(=O)C(C)(C)OC(C)C)C1 N1(C(c2cc(C)n(C)n2)=O)CC2(CCC2)CC1C(=O)NC1COC(C(C)C)C1 c1(NC(C2CCC(CNC(COCCOC)=O)CC2)=O)n[nH]c2ccccc12 C1(NC(C(COC)CC(C)C)=O)CCN(C(c2n[nH]cc2Cl)=O)CCC1(F)F Cc1c(C(=O)NC(CNC(=O)C(C)(C)C2CCCO2)C2CCC2)cnn1CCO N1(C(C(CC(N)=O)NC(=O)CC2CCCC3CC23)=O)CCC2(CNC(=O)N2)C1 N1(C(Cc2c(C)ocn2)=O)CCOC(C(N2CCN(CCO)CC2C)=O)CC1 c1(C(=O)NCCC2N(C(CC(C)C(F)F)=O)CCSC2)cccc2nn[nH]c12 N1(C(C2CCC(C)(C)CC2)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C=CI C1(NC(C2(C(=O)NC)CCCC2)=O)CN(C(=O)CCC(C)(C)OC(C)=O)CC12CC2 c1(OC)cccc(CC(=O)NCCCN(C(=O)COc2cccc(C)c2)C)c1 Cc1ccc(Br)c(C(N2CC(CNC(C3C(C)(C)C3(F)F)=O)C3(CC3)C2)=O)c1 S(=O)(=O)(c1ccc(N2CCC(CC3CCCCC3)CC2)nc1)N(CC(C)CO)C C(c1ccc(O)cc1)=CC(N1C(CCNC(c2c(C)scc2)=O)CCCC1)=O c1(C(=O)NCCC2N(C(C3(C)CCOC3)=O)CC(F)(F)C2)ccc2ncsc2c1 c1(OC)ncc(C)c(C(=O)NC(C)C(C)NC(=O)Cc2ccc(F)c(F)c2)c1Cl c1(C(=O)NCCC(C)CC(=O)NC2CC3(C2)CC3(F)F)occ2c1CCC2 c1(NC(CCCC=C)=O)ccc2c(c1)CCN(Cc1cc3cccnc3[nH]1)C2 C1(C(=O)NCC(NOC)=O)C(C)CCN1C(=O)Cc1nonc1C CC(C#N)CCC(=O)N1CCOC(C)(CNC(c2ncc[nH]c2=O)=O)C1 CCCCC(O)C(=O)N1C(CC(N2CCCCC2CCOC)=O)C2CCCC12 CN1C(=O)CN(CC2NC(=O)COC2(C)C)CC1=O C=CCC(CC)C(=O)NCC(=O)NCc1nn(C)cc1CC1CC1 c1(C(=O)NCC(C)N(C(C=CC(C)(C)SC)=O)C)cnn2c1CN(C)CC2 C1(NC(CC2OCC(C)(C)C2)=O)Cc2ccccc2C1NC(C1CCC1(F)F)=O O=C1NCc2c(C(=O)NC34CC3CN(C(=O)C(Cl)(Cl)Cl)C4)cccc21 C=CCCC(F)(F)C(=O)N1CC2CC1CC2CCNC(C12CCC(CC1)CC2)=O C(CC(O)C(=O)N(CCNC(C1CC12CC(O)C2)=O)CCc1ccccc1)SC C1(C)(CC)CCCN(C(=O)COC2(C)CN(C(C3CN(C)C(=O)N3)=O)C2)C1 C1(C(=O)NC(C2CCN(C(c3sc(C)c(O)n3)=O)C2)(C)C)CC2(CCOC2)C1 C12(C(=O)NCc3c(C)n[nH]c3)CCN(C(c3[nH]ccc(=O)c3C)=O)CCC1C2 c1(C(N2CCCC2c2ccncc2)=O)cc(F)c(F)cc1Br.c12ccc(cc1)s2 O=C1Nc2ccc(Br)cc2CCC1Sc1ccc(Cl)cc1 c1(C(N2CCC(O)(c3cn(CC(=O)NCC)nn3)C2)=O)cc(F)cc2c1CCC2 C(C)(CCC(=O)NC(C1CCOC1)(C)C)NC(c1ccc(CC)o1)=O Cc1nc(NCCN(C)C(=O)NC(C)C2CC2)c(C)c(O)n1 c1(NC(c2c(-n3ccc(C)n3)cccc2)=O)nc(C)ccc1F C1(C(=O)Cc2cn(C3CCC(NC(CN4CCC(OC)C4)=O)C3)nn2)NC(=O)NC1=O C1(NC(CSCCC)=O)CC(C(=O)N(CC(C)C)CC2CC2)C1 C(CNC(=O)CN1CC2CC2C1)(C(=O)NC1CCN(C(N)=O)C1)N(C)C c1(C(=O)NCC2CC(F)(F)CN2C(=O)C2CC2)ccc(F)c(Cl)c1F C=CC(CC)CC(=O)N1CCC(N=[N+]=[N-])(C(=O)NC(C)CN(CCCC)C)C1 N1(C(CCCC#N)=O)CCCC(C(=O)NCC2CC(c3ccccc3F)C2)CC1 c1(OC)csc(C(N2CCN(C(=O)CC3CCCC3)CC2)=O)c1OC C(=O)(C(C)CC(=O)N1CCC(F)(C(=O)NCCN2CCCC2)CC1)OC c1(C(=O)NC2CC(F)(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)ccc2cccnn12 c1(OC)cc(C#N)ccc1NC(c1cc(F)c(C)c(Br)c1)=O C1(NC(C(c2c[nH]c3ccccc23)C)=O)CC2CCC1N(C(=O)CC1CC1)C2 c1(C(N2CCC(C(C)NC(Cc3cc(C)sc3)=O)C2)=O)cc([N+](=O)[O-])cnc1C c1(C(=O)OCC)nc(=NCC2CC(NC(c3ccc(SC)s3)=O)C2)cc[nH]1 Cc1cc(C)c(OCC(N2CCC(C)(CNC(=O)CC3CC3(C)C)C2)=O)c(C)c1 N(C1CCOc2ccccc21)C(=O)NCc1cccn2nccc12 c1(C(N(CCCCN(C(=O)CCCC(N)=O)C)C)=O)ncc(C#N)cc1Cl Cc1ccc(OC2CC(NCCNC(NC(=O)NCc3nc(C)nn3C)=S)C2)cc1 C1(NC(C(C)Sc2ccccc2)=O)CC2CC(C1)N(Cc1csnn1)C2 C(=O)(C(C)N(OC)C(=O)C1C=CCN(C(=O)CC2CC(=O)NC2=O)C1)OC C(c1ccc(OC)cc1)=CC(=O)NC(CNC(C1(COC)CCC1)=O)CO C1(NC(C(C)(C)C)=O)CC(F)CN(C(C2CC3C=CC2C3)=O)C1 CC1CCCN(C(c2ccc(N)c(F)c2)=O)C1CNC(c1cscc1C(F)F)=O c1(C(C(=O)N(C)CCNC(c2cc(Br)co2)=O)=O)cnn(C(F)F)c1 N1(C(=O)NC2CCN(c3ccc(OC)cc3)C2)CC2C=C(Br)C2C1 c1(OC)ccc(CC(=O)NCc2ccc(-c3ccccn3)cc2)nc1 Cc1c(Br)cc(OC(=O)CCCn2ccnc2)cc1[N+](=O)[O-] C(=O)(C1CNC(=O)c2ccnn21)NC1CC(NC(c2c(OC)ccc(C)n2)=O)C1 c1(CC)c(C(=O)NC(CNC(=O)C=C2CCC2)C(C)C)[nH]c(C)c1C(=O)OC C1(CC(=O)NC2C(C)(C)C(OC)C2(C)C)COc2ccccc2O1 Cc1c(C=CC(N2CCC(CNC(c3sccc3Br)=O)C2(C)C)=O)cnn1C C1(CN(C(C2CCN(OCC)C2)=O)CC)CCC(Nc2n[nH]c(C)n2)CC1 C(=O)(CS(=O)(=O)c1ccc(Br)cc1)N(C(C)C)CCNC(C1CC1(F)F)=O c1(C(=O)NCC=CCNC(C2CC2C(F)(F)F)=O)cc2sccc2s1 CC1=NOC(C)(C(N2CCC2CNC(C2(c3cnn(C)c3)CCCO2)=O)=O)C1.N C1(F)(CNC(c2cn(C(F)(F)F)cn2)=O)CCCN(C(=O)C=Cc2cncs2)C1 Cc1cccc(C(F)C(N2CCSCC2CCNC(=O)CC2CC2)=O)c1 Cc1[nH]nc(C(N2CCC(NC(=O)N(C)C)CC2)C(=O)NCC2CCOC2)c1Br OCCC(N=c1ccnc(NCC(Cc2ccoc2)CO)[nH]1)c1ccoc1 Nc1ccc(Br)cc1C(=O)NCC1CCCC(NC(=O)Cc2cccnc2)C1 c1(NC(CCOCCNC(c2cnn(CCO)c2)=O)=O)ncccc1O N1(C(C(C)n2ccnc2)=O)CCC2(CC1)CN(C(C1CC(O)(C#N)C1)=O)CCO2 N1(C(CC2(C)N(C(CC(C)C3CCCO3)=O)CC2)=O)CC(F)(F)C1C1CC1 C1(CNC(C2CCc3c[nH]nc3C2)=O)CN(C(=O)C2=CCC2)CCC12CCC2 NCCC(=O)NNC(=O)NC1CCC1c1ccc(F)c(F)c1 CC1(C(=O)NCC23CC2CN(C(c2ncc[nH]c2=O)=O)C3)CCCCCCC1 C1(NC(COC)=O)CC2(CCCCN2C(c2cccn2Cc2ccccc2)=O)C1 CCC(O)C(C)C(=O)N1CCC(C)(CNC(C23CC2C3)=O)CC1 CC(C)C(C(=O)NCC1CCCCC1NC(=O)Cn1ncccc1=O)C(C)C CC(C)C(C)(O)C(=O)NC(c1nc(C(=O)N(CC(F)F)C2CC2)co1)C Cc1cc(C(C)NCC2(O)CCC2C)ccc1C#N C(=O)(CS(=O)(=O)CC(C)C)O.C=CCC(CNCCC)C(=O)OC N1(C(CCOCCN(C(=O)CN2C(=O)CNC2=O)C)=O)CC(F)CC1CO Cc1cc(N)ccc1C(=O)NC(C1CCCCN1C(=O)Cn1ncccc1=O)C c1(CSCC(=O)NCC(CNC(C2(CC)CCCC2)=O)O)cccc(C)c1 CN1C(=O)CCC1C(N1CCC(CCNC(c2cccc(C(F)F)n2)=O)C1)=O Cc1ccc(O)cc1NC(C1(CNC(=O)C=CC(F)(F)F)CCCC1)=O c1(C(N2CCC(c3ccc(C)s3)CC2)C(=O)NCCC#N)ccc2c(c1)CCC2 Cc1ccc(C)n1CCC(=O)NC1(CCCC(=O)N2CC(N3CCCC3)C2)CC1 C(=O)(C(F)(F)CCc1ccccc1)NC(CC)(CNC(=O)CCOCC(F)F)CC C(=O)(C1=NOC(C)C1C)NCC(C(=O)NC(CC)(C)C)O C1(C(=O)NCCCC(=O)N(C)CC2(OC)CCCC2)(OC)CCCCC1 C1(C(N2C3C(NC(c4ccc(CN(C)C)[nH]4)=O)C(C3)C2)=O)CC2(C1)CC1(CC1)C2 c1(SC)ccc(Cl)c(C(=O)NC2CC(O)(CNC(=O)CC3CCCS3(=O)=O)C2)c1 CCC(C)C(O)C(C)C(=O)N1CC(C(=O)N(CC(C)(C)O)C)C(C)(C)C1 N1(C(C(C2CCC2)OC)=O)CCSCC1CCNC(=O)C(C)(C)c1ccn(C)n1 C(C(=O)Nc1ccc(Cl)cc1F)(C1=NOCC1)N1CC(C)OC(C)C1 c1(C(C2C(O)C(O)CN2C)NC(C(C)Oc2ccccc2)=O)cc(Br)ccc1F C1(NC(=O)N(c2cncs2)CC=Cc2ccccc2)CC2CC1C(O)C2O CN1CC(C(=O)NCC(C)(CO)NC(c2cc(O)cc(O)n2)=O)CCC1=O CC1CC=C(C(=O)N2CCN(C(c3cc4ncccc4o3)=O)CC(O)C2)CC1 CCC(CC)(C(=O)N1CC2CCC(C(=O)NC3(C)CCSC3)(C2)C1)C(C)C C(=O)(C1=CC2CC(C1)CC2O)N1C(CCNC(C(CCC)CC)=O)CCC1 C1(CC(=O)NCC(CN(C(CC(CC)SC)=O)C)(C)C)CCC(F)(F)CO1 N1(C(=O)OC(C)(C)C)CCC(NC(c2ccc(F)c(F)c2)=O)C(F)(F)CC1 c1(CCC)cccc(NNC(=O)NCC2CCCC(NC(=O)OC(C)(C)C)C2)c1 CC(C)C(C)(O)C(=O)NC1CCN(C(=O)CC2CC(=O)NC2=O)CC1 CCCCC(F)C(=O)N1C(C(=O)NC)CC1C.C12(CC1)C(=O)NC2 CCC(CC(=O)N1CC2(CCN(C(C3CN(C)C4(CCC4)C3)=O)C2)C1)C(C)C C1(O)(CC2(C(=O)NCCN(C(=O)Cn3cc(C4CC4)cn3)C)CCC2)CCCC1 C(=O)(C1CCc2c(Cl)cccc21)NC1CC2(C(NC(C3CC4CCC3O4)=O)C2)C1 N1(C(c2cccc(COC)c2)C(=O)Nc2ccccc2)CCS(=O)C(C)(C)C1 C12(C(N3CCC(=C)C3)=O)CC(CN(C(C3CCCSC3C)=O)C1)C2 N1(C(CC2CC(C)C2)=O)C2CCC1CN(C(c1cc(C3CC3)ncn1)=O)CC2 C(=O)(C(C)(C)Cc1cnn[nH]1)N(CCCCNC(c1cc(C2CC2)on1)=O)C C(=O)(C(CC)CCCC)N1CCC(CNC(CC=CC)=O)(CO)CC1 N#Cc1ccc2c(c1)CCCC2Nc1cc(N2CCC(O)C2)ncn1 C(=O)(C(C)S(N)(=O)=O)NCC1N(C(CN(C(C)C)C)=O)CCCC1 CN1CCN(C2CC(CNC(c3ccc(CC(F)(F)F)cc3)=O)C(O)C2)CC1 Cc1nc2c(N3CCCC4(NC(C5CC5(Cl)Cl)=O)CC4C3)ncnc2s1 C(=O)(CCCC(F)(F)CO)N1CC(O)(CNC(COC(CC)(C)C)=O)C1 C1(NC(c2cc(C)[nH]c2)=O)CCC(N(c2ccc(C(F)(F)F)cn2)C)CC1 c1(OC)csc(C(=O)N(CCCCNC(c2cc(CC3CCC3)c[nH]2)=O)C)c1 c1(OC)cc(Cl)c(C(=O)NCC2CN(Cc3ccc(OC)nc3)C2)cn1 CC(C)C#CC(=O)NC1(C(F)F)CC(NC(=O)CCCC2CCCO2)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)C(c1ccc(-c2ccc(F)c3occc23)nc1)=O c1(OC)cccc(COC(C)C(=O)N(CC(C)NC(c2cnccc2Cl)=O)C)c1 c1(C(CC)C)ccc(C(=O)NCC(C)CN(C)C(C2COC(=O)C2)=O)cc1 C1(C(=O)NC2CCC(N(C(=O)CSC3CC3)C)CC2)OCC2COCCC12 CN1N=C(CC(=O)N2CC(C(=O)N(C)CC3(O)CCOC3)CC(C)(C)C2)CC1=O N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)(CNC(c2cnc(C)[nH]2)=O)C1 C1(C(=O)NCC2C(NC(CCc3scc(C)n3)=O)C2)CC2C=CC1C21CC1 c1(C(=O)NC2CN(C(C(n3cnc(C#N)n3)C)=O)C2)ccc(F)c(C(C)(C)F)c1 N1(C(c2oc(CC)c(C)c2)=O)CCC(CC)(NC(=O)C(O)C(C)SC)CC1 C(=O)(C(CC(C)C)N(C)C(c1cc(C(N)=O)co1)=O)NCC(C#C)C(C)C Cc1ccn(CC(=O)NCC2CCN(C(C3CC4C=CC3C4)=O)C2(C)C)c(=O)c1 N1(CC(c2ccccn2)(C)C)CCC2(CC(=O)NC2=O)C1 C(=O)(CCCC(C)=O)NC(CNC(C(CC)(C)F)=O)C1CC1 Cc1nc(C=Cc2nnc(SCC(N)=O)o2)[nH]c1C N1(C(C(COCC)n2cc(CN3CCCC3)nn2)=O)CCCC(O)(CC)C1 C1(NC(C2(COC)CCOCC2)=O)COCCN(C(C2(C)CCOC(C)C2)=O)C1 N#Cc1ccc(=NCC(=O)NC(CNC(=O)CCC(F)(F)F)CO)[nH]c1 C=CCCCCCCCC(=O)NC(C)C(C(C)C)NC(c1ccc(C)c(N)c1)=O C1(C(=O)NCC(=O)NCCO)(Nc2ccco2)CCC1.C1(=O)C=CCN1C1CC1 c1(N2C(C)CC(CNC(C3(COCC)CC3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] C(C1(C)CCOCC1)=CC(=O)NCC(N(C)C(c1ccnc(O)c1)=O)C1CC1 N1(C(C(CC)NC(C)=O)=O)CC(C)(C)CC1CNC(c1cn(C)nc1C(C)C)=O c1(C(=O)NCC2(C)CCCN(C(c3cccs3)=O)C2)ccnc2[nH]cnc12 Cc1ccc(C(N2CC3(NC(c4scnc4Cl)=O)CC2C3)=O)c(F)c1F CC1CN(C(C2CCCC2O)=O)CC1C(=O)NC(CC1CCCC1)CO c1(OC)cnccc1C(=O)NCC(O)CN(C(=O)CC1CCCC12CC2)C C1(C2CN(C(c3cccc(C)c3N)=O)C2)(NC(C2CC(CC)C2)=O)CC1 C(CCCCC(=O)N1CC2CC(NC(c3cnn(C4CC4)c3Cl)=O)C1C2)OC CC1=C(C(=O)N(C)CC2CCCN(C(c3c(C)[nH]c(C)c3C)=O)C2)CCO1 C1(CC)CC(C(N2CCCC(CC3CC3)C2)=O)CCN1C(=O)CNC(=O)OC C1(OC)CCCN(C(=O)C(=O)Nc2cccc(Cc3nc(C)cs3)c2)C1C C(=O)(C1=C(Cl)CCC(C)C1)NC(CC)CN(C(=O)CCN1CCCCCC1)CC C1(C(=O)NC2CCC(C(C)(C)C)C2)CC2CC1(c1cccc(C(F)(F)F)c1)C2 c1(C(N2CCC(NC(c3c(C)coc3)=O)C2)=O)cc2c(Cl)cccc2s1 C1(NC(C2(C#N)CCCC2)=O)CN(C(c2ccnnc2)=O)CC2(CCC2)C1 C#CCC(C)(C(=O)NCCN(C)CC=C)NC(=O)CC1COCC1O Cc1ccc(F)c(C(=O)NC2CC(NCc3ccc(C)s3)C2)c1 c1(OC)cc(C(N2CCCN(C(c3cc(Br)oc3C)=O)CC2)=O)cc(C)n1 N1(C(C(C)OCCOC)=O)CCN(c2cccc(C)c2)CC1.C(CN(C)CCF)N C(=O)(CCCC(=O)NC(C)CCCNC(C1CCN1C1CCCC1)=O)OC Cc1cc(N2CCCC2CN(C(=O)C(C)Oc2ccccc2)C)nc(C)n1 c1(OC)nccnc1C(=O)NC(c1ccccc1)CNC(c1csc(CO)n1)=O N1(CC#C)CCCC1C(N1CC(C(C)NC(=O)C(c2cscn2)N(C)C)C1)=O C1(NC(C=CC)=O)(CC)CCCN(C(=O)C(C)SC)C1 C(CC(=O)NC12CC1CN(C(c1cc(C)n(C)c1C)=O)C2)(C(N)=O)NC(C)=O C(CC(=O)NC1(CNC(=O)CC2CCSC2)CCC1)N(C)CCO N1(C(C(C)(C)NC(C(c2ccc(C)cc2)N(C)C)=O)=O)CCOCC(C)(C)C1 CCN(C(C)C)N(Cc1ccccc1OC(F)F)C1CC1 c1(C(=O)NC2CC(CNC(C(c3cccc(F)c3)C)=O)C2)ccc(C(F)F)cn1 C1(C(N2CCOC(CNc3ncccn3)C2)=O)CCC2(CC2)C1 N1(CC=C)C(=O)NC(c2cnc(OCC3CC3)s2)C(C(=O)OCC)=C1CCCCl N1(C(c2c(C)ccnc2)=O)CC(C(=O)N(CC(C)O)C)CC1(C)C c1(CCC)nc(C(=O)N(CCC(C)NC(C2CCCOC2)=O)C)cs1 N1(C(c2cc(Cl)ncc2Br)C(=O)NC(C(=O)OC)C)CC(C)S(=O)C(C)C1 C1(c2nnnn2C2CCC2)(Nc2c(COC)noc2)CCN2CCCCC12 N1(C(C2(C#C)CC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C(C)C1 C(=O)(CC(C)P(C)(C)=O)NCCCNC(c1c(OCC)cnc(Cl)c1)=O CS(=O)(=O)C1CN(C(=O)C(O)C2CC2)CC1NC(c1cc(-c2ccco2)no1)=O N1(C(c2c(C)ccc(C)n2)=O)CC(NC(=O)CC2CCC2(C)C)C2(CCC2)C1 C1(NC(c2c(C)csc2)=O)CCC2(CC1)CN(C(c1cnnn1C)=O)C2 N1(C(Cc2nc(COC)sc2)=O)CC2(CCCN(C(=O)C(F)n3ccnc3)C2)C1 Cc1ccc(CN(C(c2ccc(CO)c(F)c2)C(=O)NC2CCCC2)C)cc1Cl N1(C(C=CSC)=O)C2CCCC1CC(NC(C1CCCC3(CC3)C1)=O)C2 C1(NC(C(C)NC(c2ccco2)=O)=O)(CO)CCN(C(=O)CCCNC(N)=O)C1 C1(C)(C(=O)NC2CN(C(CC(CCC)(C)O)=O)CC2C)Cc2ccccc2C1 Cc1cc(C(=O)NCC2(C)CCC(NC(=O)C(C)C(F)F)CC2)cc(C)c1C c1(C(N2CCC(O)(CCNC(C3CCC3)=O)C2)=O)nnn2ccccc12 C1(C(=O)NCCC2(NC(=O)C3=CCCCO3)CCC2)CCn2c(O)nnc2C1 C#Cc1ccc(C(=O)NC(CN(C(=O)CC2CNC(=O)C2)CC)CC)cc1F c1(CCC(=O)N(C2CCN(C(c3ccco3)=O)C2)CCO)ccc2c(c1)CCO2 N1(C(CSc2cn(C)nc2)=O)CC2(NC(c3cn(C(C)(C)C)cn3)=O)CCC1C2 c1(C(=O)NC2(C(=O)NCC)CC2)cnn2c(C)cc(C)nc12 C1(C)(NCC(=O)NCCC=CCNC(C(c2cccc(Cl)c2)C)=O)CCOCC1 CC1(C(=O)NCC2CC(O)CN2C(=O)C=Cc2ccccc2Cl)CC2CCC1C2 C(=O)(C(CCC(C)C)NC(C)=O)NCCC1(OC)CN(C(c2cnco2)=O)C1 c1(OC)cccc(C2(C(=O)NCC(C)(C(C)C)NC(C3C4CC5C(C4)C35)=O)CC2)c1 c1(NC(C)=O)cccc(C(=O)NC2CN(C(c3cc[nH]n3)=O)CCC2F)c1C c1(C(=O)NCCN(C(CC(=C=C)C)=O)C)ncc(F)c2ccccc12 c1(C(=O)NCC2CN(C(CCNC(=O)CO)=O)C2)ccc(-c2ccncc2)cc1.CO CC1C(NC(c2csc(C(F)F)n2)=O)CCN1C(C1CC(F)(CO)C1)=O C1(C(=O)NCC(c2nc(C3CCC3)cs2)N(C)C)CCCC1(C)O C1(NC(CCN(C(C(C)SCCCC)=O)CC2CC2)=O)CCCC1(C)O N1(C(c2cn(CC=C)nn2)=O)CCC(F)(C(=O)NCC(CO)OC)CC1 C(=O)(C1CCc2cccc(O)c21)N1CC(N(C(C(C=C)O)=O)C)C1 CCC(C)CC(C)C(=O)N(C(C)CNC(c1ccc([N+](=O)[O-])cc1)=O)C N1(C(=O)COc2ccccc2)CC(=O)NCC1C(N1CCSC2(CC2)C1)=O C1(NC(c2ccc(C)nc2N)=O)CN(C(=O)COC2(C)CCC2)C2(CCC2)C1 c1(CC(=O)NCCC(C)N(C(C(CSC)OC)=O)C)c(C)nc(C)nc1O c1(C(=O)NCC2OCCN(C(C(CCN(C)C)O)=O)C2)cccc(C#CCO)c1 N1(C(CCNC(=O)OC)=O)CCC2CC1CN(C(C1(F)CCN(C)CC1)=O)C2 c1(C(N2CCC(C)C2C(=O)NC2CCCC2)=O)cc(=O)n(C)cn1 CCC(O)C(C)(C)C(=O)N1CC2(CC(NC(=O)CC(C)(C)COC)C2)C1 Cc1cc(C(=O)NC2CC2CNC(C2(C(F)F)CCCC2)=O)cnc1C(F)(F)F C1(C(=O)NC2CCC(COCC)CC2)CC2CCC1N2C(C1CC12CCC2)=O C(=O)(C#CC1CCC(=O)CC1)N1CCC(C(C)C)(NC(=O)C(=O)NC2CC2)CC1 C1(C(=O)NC2C(CNC(C(C(=C)C)(C)C)=O)CCC2)CC2(CCOCC2)C1 c1(C(N2CCC(n3cnnn3)C2)C(=O)NC)ccc(C(F)(F)F)c(F)c1 C1(C(=O)NCCC2C(C)OCC2)(NC(c2cc(O)nn2C)=O)CCN(C)C1 c1(C(=O)NCC2OCCCN(C(C(CC(=C)C)C)=O)C2)cc(C#N)ccc1O CC(C)(C)CC(O)CC(=O)NCCNC(c1ccc([N+](=O)[O-])c(C(N)=O)c1)=O FCC(C(F)(F)F)c1nc(-c2cscn2)nn1CC(F)(F)F Cc1cn(CC(=O)NCC2CC(O)(CNC(=O)C(Cl)=CCl)C2)c2ccccc12 S(=O)(=O)(c1ccc(NC2CN(C)C2)c(Br)c1)N1CC(CC)OCC1C N1(C(C(CC(C)C)ONC(=O)CC2CC=CCC2)=O)CC2(C)CC1CCO2 c1(CNC(C2(CNC3CCCO3)C(C#C)C2)=O)cc(OC)cc(OC)c1 C(=O)(C1=CCCOC1)N(C1CC(C)CN1c1ncc(Oc2ccccc2)cn1)CC N1(C(c2ccc(OCC)cc2)=O)CC(NC(c2coc(N(C)C)n2)=O)CC1(C)C CC(O)(CNC(c1cn(CCC2CC2)nn1)=O)CNC(c1cn(C2CC2)cn1)=O C1(C)(NC(CCN2CCN(C)CC2)=O)CCN(C(C2COCCO2)=O)CC1 n1(CC(=O)N(C)CC2CN(C(CCCSC)=O)CC23CC3)nc2c(n1)CCCC2 CC1=NOC(=O)C(CC(=O)NC2CCCC2NC(c2cccc(C(F)F)n2)=O)C1 c1(-c2cn(C(C)CNC(=O)CO)nn2)ccc(C(F)(F)F)cc1 C1(C(=O)Nc2ccc(C)cc2O)C2C(CN1Cc1cc(O)cc(O)c1)C2(C)C c1(NCC(C)N(C(=O)CSc2nncn2C)CC)ccc([N+](=O)[O-])cc1C CC1CC(C)N(C(c2cccc(C(F)F)n2)=O)CCN1C(=O)CS(C)(=O)=O C(C(C)(C(C)C)NC(C12CSCC1C2)=O)NC(c1c(C)nns1)=O c1(SCC(=O)NCCC2(CNC(C(F)OC)=O)CC2)nnc(S)s1 CCC(CC)(CN(C)C)C(=O)NCc1ccncc1Cl c1(C(=O)NCC(CNC(C2CC2F)=O)OC)ccc2nc(C)n(C)c2c1 c1(C(C(=O)NCCCOC)N(c2cc(C)ccc2F)C)cc(OC)cc(Br)c1 Cc1nc(C(N2CCCCC2CNC(=O)Cc2cc[nH]c2)=O)c(Br)s1 CC1(C)CCN(Cc2cn(-c3cccc(Br)c3F)nn2)CCS1 c1(C(N2CCN(C(C(CCC)C)=O)C(CC)C2)=O)cc(O)c(O)c(O)c1 Cc1ccc(CC(=O)N(C)CC2CN(C(=O)CSCCC#N)CCO2)cc1 c1(C(=O)NCC(C)(C)CCNC(c2cnn[nH]2)=O)cc2cccc(Cl)c2s1 C=C(Cl)CCC(=O)N(CCC(C(C)C)NC(c1cscc1-c1ccccc1)=O)C c1(C(=O)NC2CCN(C(C3(C)COCCO3)=O)CC2O)ccc([N+](=O)[O-])cc1Cl C1(NC(CCOCC)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CC2(CC2)C1 C1(C)(CC)CCC(C(N2CC=CC2C(=O)NC2COCC2N(C)C)=O)O1 c1(C(=O)NC2CN(C(CS(CC)(=O)=O)=O)CC2O)cc2cc(Cl)ccc2o1 C1(C(=O)NCC2C3CN(C(c4cc[nH]n4)=O)CC23)CCOCC12CCC2 N1(C(CC(C=C)C)=O)CCCC(N(C)C(c2ccc(CCO)cc2)=O)CC1 c1(C(N2CC(CC=C)(NC(C3CC4C=CC3O4)=O)C2)=O)ccc(Br)c(C)c1 N1(C(C(C)NC(N)=O)=O)CCC(O)(CNC(C23CCN(CC2)CC3)=O)CC1 C(CCN=c1[nH]ccc(=NC(C)C(C)CO)[nH]1)N(S(NC)(=O)=O)COC CN1CC(O)CCC1C(=O)N(CCC(=O)NCCC1CCCCO1)C1CC1 N1(C(C(CC(C)C)C)=O)CC23CCCC2(C1)CN(C(c1occc1Br)=O)C3 C1(NC(C2OCCC(=O)C2)=O)CN(C(=O)CCc2ccoc2)C2CCCC12 N1(C(c2cn(C)c(O)n2)=O)CC2CCN(C(=O)CCCCCF)CC12 c1(C(N2CCC(NC(C3(CCC)CC3)=O)C(C)C2)=O)n[nH]c2c1CCSC2 C(=O)C=CS(=O)(=O)CC.C1(CC=C)CCCCN1C(C1OCC1(C)C)=O N1(C(C2(CNC(c3ccc(CCO)o3)=O)CCCO2)=O)CCOC(CF)C1 Cn1cc(CC(=O)NCC2CCCC2NC(=O)Cn2cnnn2)cn1 N1(C(C(C(C)C)NC(=O)OC)=O)CC2CCN(C(=O)Cc3cnc[nH]3)C(C2)C1 CC1ON=C(C(=O)N2CC(NC(c3c(F)ccc(O)c3F)=O)C3CC3C2)C1C CCCC(CCC)C(=O)NC1CC(CCNC(C2CCCCO2)=O)C1 N1(C(C(C2CC2)OCC)=O)CCC2CCN(C(C3COCC(C)(C)O3)=O)C2C1 c1(Cc2ccc(C)o2)nc(-c2ccc(Cl)cn2)nn1-c1nc(Br)nn1C N1(C(COC)=O)CC(F)(F)CC1CCNC(=O)C(C)Cc1ccco1 Cc1ccc(Cl)c(C(N2CCC(C(C)(C)CNC(C3COC(C)C3)=O)CC2)=O)c1 N1(C(c2n(CCC)ccc2)=O)CC(NC(C2CCCCCS2(=O)=O)=O)C2(CC2)C1 Cc1cccc2c1CN(C(C1CC(O)CN1Cc1c(F)cccc1Br)=O)C2 c1(C(=O)NCC(=O)NC(N2CCc3ccccc32)=O)n[nH]c2ccc(F)cc12 c1(C(=O)NCC2N(C(CC=C(C)C)=O)CCCC2C)cc2ncccc2[nH]1 N1(C(C2CCC=CCC2)=O)CCOCCC1Cn1cc(C2CC3CCC2O3)nn1 N1(C(C(F)=CCC)=O)CCCC(C2CN(C(c3ccn(CC4CC4)c3C)=O)C2)C1 c1(OC)cccc(C(N2CCN(C(c3ccc(C)c(F)c3)=O)CC2CO)=O)c1N Cc1ccc(F)c(C(=O)NCC#CCNC(=O)CC2=CCCC2)c1O c1(C(N2CC(CNC(C3N(C)CSC3)=O)OCC2)=O)cccc2c1COCC2 c1(NC(C2(NC(C3CCCC(O)C3)=O)CCC2)=O)ccn2nccc2c1 c12c(C)nc(nc1O)SCC(=O)CC2.c1(CC(COC)CO)ccc(F)c(F)c1 C1(NC(c2cnn(C)n2)=O)CC2CCC1(N=c1[nH]nc(C3CC3)o1)C2 C1(C(N(C)CC2CCN(C(C3(CC(C)C)CC3)=O)CC2)=O)CC2CCCCC2O1 C1(NC(C(CCC)C)=O)CC(O)CN(C(=O)CCc2cccnc2F)C1 C1(NC(c2cccc(F)c2F)=O)CCN(C(C2(C3CCCO3)CC2)=O)CC1C(N)=O C(C)(N=c1nc2c(ncn2C(C)C)c(NCc2ocnc2C)[nH]1)c1c(C)nns1 C1(CNC(CCNS(C)(=O)=O)=O)CCN(C(=O)C(C)(C)C#N)CC1 C(=O)(C(O)C(C)(C)CC)N1CCN(C(C2(OC)CC2)=O)CC1C(C)C C1(C(=O)NCC2CCN(C(c3n(C(C)C)ccc3)=O)C2)CCS(=O)(=O)C1(C)C CC1(C)CCCC(CC(=O)NC2CC(C)(NC(=O)CSCc3ccncc3)C2)O1 C1(C(CNC(=O)C(F)=CC2CC2)F)CCN(C(C2CC3C=CC2C3)=O)CC1 c1(NC(C2CCN(C(=O)NC(c3ccccc3)C)CC2)=O)cc2ncsc2[nH]1 N1(C(C(=O)NCC)=O)CCN(C(c2ccn(CC)c(=O)c2)=O)CC1CCNC CCC1(CNC(=NCCCC(C)C)NCc2cccs2)OCCc2ccccc21 Cc1ccc(NC(=O)CSCC(=O)NC(C)CC2CCCC2)c(I)c1F C1(CC(=O)NCCC(C(C)C)OCC(=O)NC2CCOC2)CCC(C)(C)CO1 Cc1cc(=NCC(C(C)C)N2CCC(C)CC2)[nH]c(=NCc2nc(Br)cs2)[nH]1 Cc1cccc2c(C(=O)NC3CC(CNC(C4CC=CCC4)=O)C3)n[nH]c12 CCCCCCCCC(=O)NC1CN(C(c2coc(C)c2)=O)C2CCCC12 C(C(=O)NCc1ccsc1C(=O)NCc1nn[nH]c1C(C)C)(C(C)C)SC N1(C(C(C(CC)O)C)=O)CCC2CN(C(c3cc4nc(C)sc4[nH]3)=O)CC2CC1 c1(C(N2CCC(OCCN3CCC3CO)C2)=O)cc2ccccc2cn1.C(CSC)O CCC(CCCC(=O)Nc1cnccc1C)NC(C1(C)CCCCC1)=O CCC(CC(F)(F)F)C(=O)N1CC(CNC(c2c[nH]nc2C2CCC2)=O)C(C)C1 C(=O)(C(CNC(C1(CCF)CCC1)=O)C(C)(C)C)NC(c1ccccc1)C c1(C(CC)C)cn(CC(=O)N(C(C)CNC(=O)C2CC2)C)nn1 c1(OC)ccc(F)c(CN2CC3CN(c4cc(C#N)ncn4)CC3C2)c1OC N1(C(c2c(OC)ccnc2)=O)CCC(C(=O)NCC(F)Cl)C1(C)C c1(CCC(=O)N(C(c2cn(C(C)CC3CC3)nn2)CC(N)=O)C)ccc(Cl)nc1 Cc1cnc(C(=O)NCC2C3CC2N(C(=O)CC2CCCCC(=O)N2)C3)cc1C CCC(C)C(C(=O)N1CC2(C)CC1(C(=O)N(C)Cc1ccoc1C)C2)N(C)C CCCCCC(CC)C(=O)N1CCC(C)(NC(c2ccc(OC)nc2F)=O)C1 N1(C(CC2C(=O)NC(=O)N2)=O)CC2(C=C(C(=O)NC3CCC(O)C(O)C3)CO2)C1 C(=O)(C(F)C(C)C)NC1(CO)CN(C(c2n(CC=CC)ncc2)=O)C1 C(=O)(C1CCCn2cnnc21)N(C1CCCC1)CCNC(C1COCCOC1)=O C(CCCCCC(=O)N1CC2(COC(=O)C2)C1)N(C)C(C1C=CCS1)=O C(=O)(C(=O)C(C)(C)C)N1CCC(N(C(c2ccc(C(C)(C)C)s2)=O)CC)C1 C12(N)CC=CC(C1)OC2.c1(NC(CN(CC)CC)=O)ccccc1.C12CC(C1)C(=O)N2 C1(SCCn2cc(CNC(COC(C)C)=O)nn2)OC(=O)CC1(C)C C12(NC(C=Cc3ccn(C)c3)=O)CN(C(=O)Cn3ncnn3)CC1CS(=O)(=O)C2 N1(C(C)=O)CC2CC2(CN(C(c2ccnn2C)=O)Cc2ccc(CO)cc2)C1 C(C)(c1ccccc1C)=CC(N1C(CNC(C2CCCSC2)=O)CC(OC)C1)=O C1(NC(C2CCC(CNC(c3c(C)nns3)=O)O2)=O)CC(=O)N(C(C)C)C1 c1(C(C(=O)NCC2N(C(COCCOC)=O)CC(F)C2)C)ccc(F)cc1F CCCCCCC(C)CC(=O)N1CCCC(C)(NC(C2CCC(C)CC2)=O)C1 Cc1cnn(CC(=O)NCC2(O)CN(CCc3scnc3C)C2)c1 c1(NC(C2(O)CCN(C(C(C=CC)O)=O)C2)=O)cc(OC)ccc1C C1(C(N2CCC(C)C2)=O)CCCCC1NC(C1(c2cccs2)CCCC1)=O N1(C(c2cnc(COC)s2)=O)CC2CC1CN2C(=O)C=Cc1cc(F)c[nH]1 N1(C(C2(SCC)CC2)=O)CCCOC(CCNC(=O)CC2CCCCC2(F)F)C1 C1(CC(=O)N(C2CN(C(=O)Cn3cc(Br)cn3)C2)C)C=CCCC1 N1(C(Cc2cc(COC)on2)=O)CC(NC(c2cscc2F)=O)C(SC)C1 c1(C(CC)(C)C)cccc(C(=O)NCCCNC(c2nnc(C)s2)=O)c1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(C3OCCCO3)=O)C2)cc1 C(Cn1cncn1)(C(=O)NOCC1CCCN1C)NC(CCN(CC)CC)=O CC(C)(C)S(=O)(=O)CC(=O)NCCC1CCCN(C(=O)C(=O)N=S(C)(C)=O)C1 c1(OC)c(C(=O)NC23CC(C2)N(C(=O)CC2(CO)CC2)C3)cccc1F N1(C(CC(C=C)c2ccccc2)=O)CC2(CCN(C(C3(C#N)CCCC3)=O)C2)C1 C(CCC(C)C)(C(=O)NC(C)C(=O)OC)N1C(CC)C(=O)NCC1 C1(CNC(C2CC3(C(NC(C(NOC)=O)=O)C3)C2)=O)Cc2nccn2C1 C(CC(CC)C(=O)N1CC(O)(CNC(=O)COc2cn[nH]c2)C1)=CC c1(OC)cc(CNc2cnc(F)cc2C(=O)N(CC(C)C)CC(C)C)c(F)c(F)c1 Cc1cc(C)c(C(N2CCCN(C(=O)C=Cc3ccc[nH]3)C(CO)C2)=O)c(S)n1 C=CCCCCC(=O)NC12CCN(C(=O)CCCCCF)CC1C2 c1(CNCCNC(C(C2CCC(=O)N2C)C)=O)c[nH]c2ncccc12 N1(C(C(CC)SC)=O)CCCC(F)(CNC(=O)C=C(Cl)Cl)C1 N1(C(CC2CC(C)C2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 c1(C(=O)NCCC(C)(C)NC(C(COCC)C)=O)cncc(C(=O)OC)c1C C1(C(=O)NCC2(O)CC(CNC(=O)CCC3CCOC3)C2)CCCNS1(=O)=O C(=O)(C(C)(F)C(F)(F)F)NC(C(C)C)(C)CNC(c1ccc(O)nn1)=O C1(CC(=O)NC2CCN(CC(=O)N(C3CC4CCC3O4)C)C2)CC(=O)NC1=O C1(CCC)CCC(CC(=O)NC(C)CC(C)NC(c2scc(C)c2Cl)=O)CC1.SCC Cc1nccnc1C(=O)NC1CCC1CNC(=O)CC1CCCN1C(C)C C12(CNC(C3(OC)CCC3)=O)CC(CO1)N(C(c1cccc(=S)n1O)=O)C2 c1(N2C(C)(C(=O)Nc3ncc(C)nc3Br)CC2)nc(Cl)c2c(ccn2C)n1 CC1(C)OCC2CC12C(=O)NC1COCCC1NC(c1csnc1Br)=O CC(CCC(C)(C)C)C(=O)N1C(C(=O)N(C2(C3CC3)CC2)C)CCC12CC2 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CN(C(=O)C(c2ccccc2)F)CC1(F)F Cc1c(C(N2CCC(OCCNC(=O)CN(C3CCCC3)C)C2)=O)ccn1C Cc1cnc2n1CCCC2C(=O)NCC(C)(C)CN(C)C(c1ccsc1)=O CCC(CC(F)F)C(=O)NCC1(NC(=O)CN2CCN(c3nccs3)CC2)CC1 C(=O)(C(C)(C)C(C)(C)O)NC1CC(CCNC(C(C)OCC)=O)C1 c1(C(=O)NC2(C)CC(NC(C(CC=CC)C)=O)C2)ccnc(Cl)c1NC c1(NC(C(N2CC3C(C)C3C2)c2c(C)con2)=O)ccccc1C c1(C2CCN(C(C(C)Cc3ccc(F)cc3)=O)CC2)cccc(C(=O)O)c1F C(C)(C)(CCCNC(c1cc(-n2cccc2)ccn1)=O)NC(COCC)=O C=CC(C)(CCOC)C(=O)N(C)CC1(CNC(=O)Cc2noc(C)c2C#N)CC1 c1(C(C(=O)NCC(C)NC(c2c[nH]nc2C(C)(C)C)=O)O)ccccc1Cl C(=O)(C1=C(Cl)CCC(C)C1)NC1C2CN(C(c3c(C)cco3)=O)C1C(O)C2 c1(N2CCN(ONC(=O)OC(C)(C)C)CC2)nccc2oc(Br)cc12 c1(CNC(CC2(C=C)CCC2)=O)cnn(C)c1C(=O)NCC1CCC(=O)N1 C1(C(N(CC(C)(C)CNC(=O)CC2CCCO2)C)=O)CCCC2(CCC2)O1 c1(CN(C(c2cc(Cl)ccc2F)C(=O)NC2CCOC2)C)nc2ncccn2n1 CCC(CC)C(C)C(=O)NCC1(CNC(c2ccnn2-c2ccccc2)=O)CC1 N1(C(CSC)=O)CCC(C2(NC(=O)CCOc3ccc(C)cc3)CC2)CC1 c1(C(N(CC(C)NC(c2cc3sccc3[nH]2)=O)CC)=O)cccc2c1OC(C)C2 S(=O)(=O)(c1cc(C)ccc1C)NC(C1CCC(CNC(CCC=CC)=O)CC1)=O N1(CCc2c(OC)cccc2)CCC(NC(C2CCC(C)(C)O2)=O)CC(C)(C)C1 C1(OC)CN(C)C(C)(C(=O)NCC2C3CC2N(C(=O)CCc2cnc(C)s2)C3)C1 CCCC(C)(O)CC(=O)NC1CCN(C(=O)C(=O)NC2CC2)C1 C(=O)(C1CCCc2nnn(C)c21)N(CC(CNC(c1onc(C)c1C)=O)O)C C=CCC(CC(C)C)C(=O)N1CC2CCCN(C(C3CCCCO3)=O)C2C1 Cc1cc(CC(N2CCC(CCC(=O)NCC3CC3C(C)C)C2)=O)no1 C(=O)(C(O)C(F)(F)F)NC1C(CNC(=O)CCCNc2ccccc2)CCCC1 N1(C(C(CC(CC)C)NC(c2ccc(C(C)C)o2)=O)=O)CCCC(C2(C)CC2)C1 N#Cc1cc(C(N2CC3(CCC(C(=O)NCC4CCC(F)C4)O3)C2)=O)ccc1Br C1(C(=O)OCC)CN(C(=O)C(C)(C)C2CCOC2)CC12CC2 C(CCC(F)(F)F)N(C(=O)CCCN(C)C(C1CCCOC1)=O)C C1(CCNCc2nc(-c3ccn(C)n3)nn2C)CCC2(CCOC2)O1 C1(OC)CC(NC(c2ccn(C)n2)=O)CN(C(=O)CC2CCCCC2C)C1 c1(C(N(C2CCN(C(C34CC(C)C3C4)=O)C2)C)=O)cccc2c1CCC2=O C1(C(NOCC(C(C)C)O)=O)CCC2CCC1N2C(=O)CCC1CC1 CC1CCCn2ncc(C(=O)NCC3CC(F)(CNC(c4cnn(C)n4)=O)C3)c21 CC1Oc2ccc(C(N3CCN(C(=O)CC4CC5(CC5)C4)CC3)=O)cc2C1C C(CN=c1[nH]c(=N)[nH]c(=NCC(C)CN2CCCC2)[nH]1)c1c(OC)cccc1C C1(CC)C(NC(=O)C(F)C(C)C)CCN1C(c1csc(COC)n1)=O C1(CC=C)(NC(C2CC23CCCC3)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC1 C1(NC(C2(CC)CCC2)=O)CN(C(c2ccc3nnnn3c2)=O)C2(CCOC2)C1 C1(NC(=O)C=CCNC(C2CCCCO2)=O)CCOC12CCCC2 c1(C(N2CCCC(N(C(=O)CC#N)CC)C2)=O)ccc(N(C)C)c(F)c1 C1(C)(C(N(C2(C(=O)NCC(C(CC)C)OC)CC2)C)=O)CC2C=CC1C2 c1(NC(=S)Nc2ccc(Br)cc2)ccc(OC2CCN(C(COC(C)=O)=O)C2)cc1 C1(NC(CC(C)(C)O)=O)CC(C2CCN(C(=O)Cc3cc(F)cc(F)c3)C2)C1 CC(C)CC(C)(O)C(=O)NCc1cc(C(N2CC(CC(N)=O)C2)=O)cs1 C1(CNC(C2CC2c2cncs2)=O)COCCN1C(=O)C=CC1CC1 N1(C(C(CSC)O)=O)CCCCC1CCC(N1CC(F)(F)C1C1CC1)=O CC1CCN(C(=O)CCc2nc(-c3ccc(Cl)cc3)no2)CC1NC(=O)CO C(=O)(CC1=CCCCC1)N1CCC(CNC(c2cc(C#N)sc2)=O)C1 CCC(CC(=O)NCCN(CCO)CC)C1CC1.C1(CC(=O)NC)CC(F)(F)C1 c1(C(N2CCC(CC)(NC(=O)C(OC)OC)CC2)=O)[nH]c2cc(C)ccc2c1C c1(C(=O)NCC(CC)NC(C2CC3(CC3)CO2)=O)cncnc1C1CC1 C1(C(N(C(C)CNC(c2cnc(SC)s2)=O)CC)=O)CC(C)=NO1 c1(-c2n(C3CCC(C)C3)nc(-c3cc[nH]n3)n2)cc(Br)c2cccnn12 CC(C(=O)NCC1CC1C(=O)N(CCCO)C1CC1)C(C)(C)C CC1CN(C(C2CC3(CCO2)CC3)=O)CCC1NC(c1cnc[nH]1)=O c1(C(N2CCC(N(C)C(C3CC4CC4C3)=O)C2)=O)ccc2c(c1)COC2 N1(CCCNC(CCN(CC=C)C(C2CC2Cl)=O)=O)CCCC1=O C1(NC(C2(C=C)CC2)=O)C2CCC(C2)C1NC(=O)CCOc1c(C)cccc1C N1(C(C2(C)CCOC2)=O)CC2(CCN(C(=O)C(N3CCCC3)C3CC3)CC2)C1 CC(C)(C)CC(C(=O)NC1(C2CCCCO2)CC1)NC(c1cccn2ccnc12)=O c1(C(C(=O)NCCCOC)N(C2CCOC2C)CC)cc(F)ccc1C c1(NCC(=O)N(C(C)C(F)(F)F)C(C2C3CNCC23)=O)nnc(O)nc1O C1(C(=O)NC2(C)CCCC2(F)F)CC2CCCC2N1C(c1ncccc1Cl)=O Cc1ncccc1CC(=O)NCC=CCN(C(C1CCCN1N=O)=O)C1CC1 C(CN=c1[nH]c(N2CCc3cncnc3C2)nc2cccc(F)c12)OCCCO CC1CN(C(c2cn(CCNC(=O)Cc3ccncc3)nn2)=O)CC(C)O1 CCCCCC(C)CC(=O)N1CC2(CCC2NC(c2cnn(C)c2SC)=O)C1 C=CCCCC(=O)N1CCCC1(C(C)C)C(=O)Nc1cncnc1C C1(c2nnnn2C2CCCC2)(N(CCCC(C)O)C)CCCCC1 C(=O)(C(C)C(CC)CC)N1C(C(=O)NCc2c(CC)noc2C)CCCCC1 C(C(C)(C)CC(=O)NC1CN(C(=O)CCC(C)N(C)C)CCC1F)OC C1(N(C(=O)CC2(C)CC(F)(F)C2)C)CCCN(C(C2(C)CC(=O)C2)=O)CC1 N1(C(CCC=C)=O)CC2(CC(NC(=O)COc3cnn(C)c3)CO2)C1 N1(C(c2c(CC)n(CC)nn2)=O)CC(O)CC1(C)C(=O)NCc1ccc(C)cc1 c1(CC(=O)NC2C3CN(C(C(C(C)C)SC)=O)C2C3)cc(C)cc(C)c1 c1(C(N(C(C)CNC(c2ccc(-c3cnn(C)c3)o2)=O)C)=O)ccc(Cl)cn1 C1(NC(C2CCCC(C)(C)C2)=O)CN(C(=O)CC2CC=CC2)Cc2ccnn2C1 c1ccn2c(=NCCN3CCc4sccc4C3)[nH]nc2c1 N1(C(C2C(c3cc(C)no3)C2)=O)CCC(O)(CNC(C23CSC(C2)C3)=O)C1 c1(-c2nnc(NC(CCC)CC(=O)OCC)o2)ccc2cnoc2c1 CON1CCC(C(=O)NCCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CCO2)CC1 N1(C(C(COC(C)C)(C)C)=O)CC2CC(NC(c3ccc(C(N)=O)nc3)=O)C1C2 N1(C(C2(COC)CCCCC2)=O)CCC(CNC(=O)CSC(F)(F)F)CC1C C1(CCC(=O)NC2(CCCNC(CN3CC(C)C3)=O)CC2)CCC(=O)C1 c1(C(=O)NCC23C(CN(C(c4scc(COC)c4)=O)C2)C3)cnc(Cl)c(N)c1 c1(C(=O)NCC#C)cc(NC2C(NCCC(=O)OCC)CC2)nc(C)n1 C(=O)(C1=C(Cl)CCOC1)NCC(CCC)NC(c1ccn(CC)c(=O)c1)=O c1(C(N2CCCC(C3CCCCO3)C2)=O)cc(C(=O)O)c2c(n1)CCCC2 N1(C(C2(NC(C(C)O)=O)CCC2)=O)CC2CC1CO2 N1(C(c2c(CC)nns2)=O)CC2CCC(N(C)C(c3ncsc3C)=O)C2C1 C1(CC(=O)NC2(C#C)CC2)CCC(C(=O)Nc2cc(C)ns2)C1 C(CCCCN(C(C1CC1c1ccccc1)=O)C1CC1)NC(c1cncs1)=O CN1CCN(C(c2ncccn2)=O)CC1CNC(C1C2CCC(F)(F)C12)=O c1(C(=O)OC)cc(N2CCC(CNC(c3csnn3)=O)C2)nc(C)n1 c1(SC2CC3CC2CN3CC2N(C(=O)NC(C)(C)C)CC(O)C2)cc2ncccc2[nH]1 CC1CC(C(N2CC(OCCN(C)C)C2)=O)N1C(=O)Cc1cncn1C c12ncnc(Cl)c1C(=O)NC1(CO)CN2C1.c1(C(=O)OC)ccnc(N(C)C)n1 N1(C(c2n(C)cnc2)=O)CCN(C(c2ccc(C(=O)C(F)(F)F)s2)=O)C2CCC12 C1(C(N(C)Cc2n(CC)cnn2)=O)C=CCCN1C(=O)CC=CC(C)(C)C N1(C(CC=C=C)=O)CCC2(CCOCC2)C(NC(=O)C(C)CCCOC)C1 c1(C(=O)OC)ccc(C(C(=O)NCC2CC2)N(C2CC2C)C)o1 C1(C2CC2)(C(=O)NC(CCOC)C(C)C)CN(C(=O)CCCN(C)C)C1 C1(NC(C2(C(C)C)CCN(C(c3c(C)ncs3)=O)C2)=O)CCCCC1N=[N+]=[N-] N1(C(C(CN(C)C)NC(C2CN3CCC2C3)=O)=O)CCCC12CCCC2 c1(CNC(=NCc2n(C)ncc2)NCCC2CCCO2)cnc(C2CC2)nc1 Cc1nn(C)c(C)c1-c1cn(CC(N2CCCC(OC3CC3)C2)=O)nn1 N1(CCCCC)CCOC2(CCN(C(=O)Cn3nc(C)c(C)c3C)CC2)C1 N1(C(c2cncc(C#C)c2)=O)CCC2(CC1)CCN(C(=O)CC1CC1C1CC1)C2 C(=O)(C1=CCC(C)(C)CC1)N1CCCC(NC(C2OCCN(C)C2)C2CC2)C1 C1(C(N(CCC)CC)=O)CC(=O)CN1C(c1cc(CC)sn1)=O C1(C(=O)NC2C(CNC(C3CCC(=C)CC3)=O)C2)CCOC2(CCOCC2)C1 c1(C(=O)NC2CN(Cc3c(F)cccc3F)CC2O)c(F)cc(F)cc1Cl Cc1nnc(O)c(C(=O)NCC2CN(c3nnc(C(F)F)o3)CC2C)c1C N=c1[nH][nH]c2ccc(-c3cnc(CC(=O)N(C4CSC4)CCN)nc3)cc12 C1(O)(C(N(C)CC2CCCN2C(C2CC3CCC2C3)=O)=O)CCCCCC1 S(=O)(=O)(c1c[nH]ccc1=NCC(CO)C1CCC1)NCCCCCC=C C#CC1(C)CCCN(C(c2ccn(CCOC)c2)C(=O)Nc2ccccc2Cl)C1 CC1(C#N)CN(C(=O)C(Cc2ccoc2)NC(c2cnn[nH]2)=O)C1 Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCCCC1NC(c1cnns1)=O c1(C(=O)NC(c2c(C)cnnc2)C)c(Cl)ccc(C)c1O N1(C(N=c2cc(C)n(CCO)[nH]2)=O)CCc2cc(F)cc(F)c2C1 n1(C(C)(C)C(=O)NCC2(NC(c3cnc(Cl)[nH]3)=O)CCOC2)cc([N+](=O)[O-])cn1 C(C)(CC(C)NC(=O)C(O)CN(C)C)NC(C1CC(CC(=O)OC)C1)=O C1(CNC(CCNC(=O)C=CCl)=O)C2CCCC1N(C(=O)C(=O)Nc1ncc[nH]1)C2 N1(C(CCCCSC)=O)CC2(C(N3CCCOCC3C)=O)CC1CO2 c1(C(N2CC=CC(NC(C3N(C)CCOC3)=O)C2)=O)cccc(C(F)F)c1Cl c1(NC(=O)NCC2C(NC(=O)CCOc3ccc(Cl)cc3)C2)cc(F)ccc1Cl C1(NC(c2ncc(Cl)cc2Cl)c2n(CC)nnn2)CCOC2(CCCC2)C1 C1(NC(CCNC(C)=O)=O)CCCN(C(=O)Cc2ccccc2C)CC1F c1(C(=O)NC(C(C)NC(=O)CCC(=O)N(C)C)CO)ncn2c1CCC2 C1(C(=O)NC(C2CCCCC2)C#C)CC2CC2N1C(=O)COCCN(C)C C(=O)(CC(C(N)=O)N(C)C)N(C(C)COC(=O)C(C)C)CC=C c1(OC)cc(N)ccc1C(=O)NCCCNC(=O)C(Cc1ccccc1)N(C)C N(C1CCc2cccc(Br)c21)C(=O)NC12CC(n3cc(CC(C)C)nn3)C1C2 C=CC(C)CC(=O)N(C)CCN(C)C(C1C(c2ccncc2)C1(C)C)=O C1(O)(CNC(Cc2cnc(C)[nH]2)=O)CCCN(C(C2CN3CCCC2C3)=O)C1 C1(O)(CN(C(CC2C(C)(C)C2)=O)C2CC2)CN(C(=O)COCC2CCCOC2)C1 C(CCC(=O)N1C(=O)CCCn2cc(C3CN(S(C)(=O)=O)C3)n2C=CC=CC1=O)OC N1(C(COCC(=O)OCC)=O)CCCCC1CCC(N1CCCC1C1(C)CC1)=O C(=O)(C(C)CC(F)(F)F)NCCCC1N(C(CCC2CC(OC)C2)=O)CCCC1 c1(C(N2CCCC(N(C(=O)CC3C(C)(C)C3(C)C)C)C2)=O)ccnn(C)c1=O CC(C)(C#N)CC(=O)N1CCC(O)(CNC(=O)COc2ccc(O)cc2)C1 C1(NC(=O)NC(C2(C(C)(C)C)CCC2)C)CCCC1C n1(CC)c(C(=O)NCC(C)(CO)NC(=O)CCCn2cccn2)cnc1O c1(CC(=O)N(C2CCN(C(C3(O)CCOC3)=O)CC2)C)ccc2c(c1)CCC2 C12(C(=O)OC)CCC(C(=O)NCCC3(O)CN(C(C4CCCO4)=O)C3)(C1)C2 c1(C(=O)NC2CC(F)(CNC(C3CCC3)=O)C2)ccc(Br)c(F)c1 c1(C(=O)NCCC2CN(C(C3COCC(C)O3)=O)C2)ccc(F)c(Cl)c1F C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCOC(C)C1C Cc1cc(CCNC(=O)OC(C)(C)C)nc(Br)c1.C12CC(F)(C1)CNC2=O N1(C(CC2(OCC)CCC2)=O)CCC(C)CC1C(=O)Nc1cccc(C(C)C)c1 N1(C(C(c2n(C)c(Cl)cn2)(F)F)=O)Cc2ccc(F)cc2C1 c1(OC)cccc(C(F)(F)C(=O)NC2CCCC2NC(=O)Cn2nnnc2C)n1 C1(NC(CCCOCCC)=O)CN(C(=O)CC2CCC(C)(C)O2)CC2CCCC12 N1(C(C2C(C)C2)=O)CC(CNC(=O)CC2=NNC(=O)C2)C2(CCOCC2)C1 N1(C(C(=O)NCC)CCC(=O)N(C)C)CCCc2cc(CC)ccc21 c1(C(=O)NCCNC(C(n2nnnc2C2CC2)C)=O)ccc(F)c2[nH]ccc12 C#Cc1ccccc1CC(=O)NCCOCCN(C)C(C1(C)CCNC(=O)C1)=O N1(C(=O)COc2cccc(F)n2)CC(NC(=O)CC23CC(C2)C3)C(CO)C1 c1(NC(=O)OCC)ccc(NC(=O)Nc2cccnc2OC)cc1C c1(C(N(CCNC(C(CO)N(C)C)=O)CC2CC2)=O)cc(O)nc(N(C)C)n1 Cc1c(CCC(N2CCC(C)(NC(=O)CC3C=CCCC3)C2)=O)cnn1C CC1CN(C(c2cc(Br)sn2)=O)CC1(C)CNC(C1(C(N)=O)CCC1)=O N1(C(CC2CC(CC)C2)=O)CC(N(C(=O)COc2cccc(C)c2)C)C(C)(C)C1 C#Cc1cc(F)c(C(=O)NC2CCN(C(=O)CN(C)C3CC3)CC2C)cc1F C1(C(=O)NCCN2CCNC(=O)C2)CC2CCN(c3cc(Cl)nc(CO)n3)CC12 C(=O)(CCCCCC(C)O)NCc1ccc(CNC(c2c(CC)[nH]c(=N)s2)=O)cc1 C1(NC(C=CC)=O)CN(C(=O)CSc2ccc(C)c(C)c2)Cc2nccn2C1 N1(C(C2(COC)C=CCN2C(=O)Cc2ccsc2C)=O)CC=C(CO)CC1 CC(C)CC(CNC(=O)C(CC1CCCC1)NC(c1ccoc1)=O)CO C1(C(N(CC)CC2CCCCO2)=O)CCC(NC(=O)Cn2cnnn2)CC1 C(N=C(NCC1CCOCC1)NC1CC(C(N)=O)C1)C1C(C)CC1 C1(C)(CNC(C2CC(C)OCC2)=O)CCCN(C(C2(F)CC2)=O)C1 C=CCC(CC)C(=O)NC1CCCC1NC(c1cc(OCC)n[nH]1)=O c1(C(=O)NCC2(C)CCC(NC(C3C(CC)C3)=O)C2)ccc(Cl)c(F)c1F CC1CC(NC(C2(C(F)(F)F)CCC2)=O)CCN1C(=O)CCC1CC1 C(=O)(C(CC(=C)Cl)NC(C1CCC(F)C1)=O)NC(C#C)(C)C O=C1OC2CCN(C(c3onc4c3CSC4)=O)C1C2 c1(OCC)ccnc(N2CCCC2Cn2cc(CNC(=O)C#CC3CC3)nn2)n1 CN1CCN(C(=O)C(C2CCCO2)NC(c2cc3n(n2)CCO3)=O)CC1CO C1(NC(CC(C)OCC2CCCO2)=O)C2CN(Cc3ccccc3)CC12 N1(CC)CC(c2nnnn2C(C)(C)C)(NC2CCNC(=O)C2)CCC1=O C1(C(N(CCCNC(c2c(C)nn(C(C)(C)C)c2)=O)C)=O)CC(C)(C)CN1C c1(C(N(CC(CNC(C(c2ccnn2C)C)=O)O)C)=O)cc2c(nn1)CCCC2 C1(C(=O)NC(CCCC=C)C2CC2)CC12CCN(C(=O)C1=CCSC1)C2 C1(C(=O)NCC(C)NC(C(C2CCCCC2)OC)=O)C(C#N)C1(C)C c1(C(N(C)CC2(CNC(=O)CCOC3COC3)CC2)=O)ccc2nonc2c1 CC1CN(C)C(C)CC1NC(c1coc(CNC(C2(C)C=CCC2)=O)n1)=O Cc1ccc(Br)cc1C(=O)NC12CC1CN(C(C1(CO)CCOC1)=O)C2 N1(C(CC2(OCC)CC2)=O)CC(NC(c2ccn(C)c2)=O)CC(O)C1 C=CCCC(CC(C)C)C(=O)N1CCC(CNC(c2n[nH]c3c2CCSC3)=O)C1 c1(CCC(=O)NC2(c3nc(COC)on3)CCOC2)cccc(C)c1C C1(C(NOCCCOC(C)=O)=O)CCOC1CNC(=O)C=NOC c1(C(=O)NC2CCCC(NC(C3N(C)C(=O)OC3)=O)C2)nccc2ccncc12 N1(C(C(CCC)OCC)=O)CCN(C(C2CC(O)C2)=O)CC1C(F)F C=Cc1cc(C(N2CCN(C(=O)C(C)=CC3CC3)CCC2C)=O)cc(F)c1 CC(CN=c1nc(N2CCC(C(C)(C)CO)CC2)c2cnn(C)c2[nH]1)C(C)(C)C c1(N2CCC(OCCNC(CCC(C)C)=O)C2)ncnc2sc([N+](=O)[O-])cc12 C1(C2CC2)(C(=O)NCC2C(C(=O)OC)CC2)CN(C(=O)C(C)N=[N+]=[N-])C1 CCCCS(=O)(=O)NCC(=O)NC(CNC(c1csc(CSC)n1)=O)CC c1(C(N2CCC(CNC(C(CC)(CC)CC)=O)C2)=O)cnc2ccc(C)cc2c1 C(c1ccccc1C)=CC(=O)NC(C)C=CC(N1CCN(C(COC)=O)CC1)=O N#Cc1cc([N+](=O)[O-])ccc1NC(c1sccc1-c1cccs1)=O c1(C(=O)NC2C3C(C)N(C(=O)CO)C2C3)cc2c(cc1Br)OCCO2 c1(N2C3CC(CN(C(C(C)OCC)=O)C3)C2)nc2ccccc2cc1[N+](=O)[O-] C12C3CN(CC13)C2=O.c1(CNC(CNC(C)(C)C)=O)cnoc1C1CCCCC1 Cc1ccc2c(C(=O)NCC3(F)COCCN(C(=O)Cc4cc[nH]c4)C3)onc2c1 c1(OCCOC(c2c(CC(=O)OC)occ2)=O)ccc(Br)cn1 CC1CN(C(=O)COC2CCN(C(C3(C#N)CCC3)=O)C2)CCN1C1CC1 N1(C(C=C(C)C(F)F)=O)CCC(C(=O)NCC2CCC(CO)O2)C1 c1(C(=O)NCCc2cn(-c3cc(Cl)cc(Cl)c3F)nn2)[nH]cc2c1CCCC2 C(=O)(C1=CC2(CCOCC2)C1)NC1C(C)CN(C(=O)CCC(=O)NC2CC2)C1 C1(C(=O)O)CCc2[nH]c(=NC3CC(N4CCCCC4)C3)sc2C1 c1(C(N2CCC(N(C(c3c(SC)n(C)nc3)=O)C)C2)=O)cccc2ncnn12 CCCCC(C)C(=O)NCC1CC(O)(CNC(c2cnc(C(C)C)nc2C)=O)C1 N1(C(c2cnc(C)s2)=O)CC(NC(=O)C(C)OCCN(C)C)C2(CC2)C1 CCCC(CNC(C1CC(=O)C1(C)C)=O)C(=O)NCc1cnc(C)n1CC C1(C(=O)NC2CC(N(C(c3c(COC)cco3)=O)C)C2)C2CN(C)CC12 C(CC1CC1)(C(=O)NC1CCSC1)NC(=O)CCC1CC1 C1(CC)CN(C(=O)CN(C(=O)COc2cc(C)on2)C2CC2)C(CC)CO1 N1(C(c2c(C)cccn2)=O)CCCN(C(=O)CC(F)(F)C(F)F)CC1C C1(C(=O)NC(C(C)C)CNC(=O)Cc2csc(Cl)n2)CC(C)(C)OC1(C)C C(CC(CNOC)NC(=O)C(F)(F)Cl)OC.C(=O)(C(C)C1CC1)NCC1CC(=O)C1 C(CCCOC)(C(=O)NCc1nc(C)c(C)o1)NC(C(CC)CC)=O C12(C(=O)OC)CCC(CC1)N(CCC(=O)Nc1cc(Cl)ccc1Cl)C2 Cc1c(C(=O)NCCC(C)NC(=O)C(C)(C)C(C)(F)F)nn2ccccc12 C(CC(C(=O)NCc1cccc(C)n1)NC(C1CC(C)=NO1)=O)OCC c1(C(N2CCC(CC(=O)NC(C34CCC(CC3)C4)C)C2)=O)ccc(O)nn1 CC(C)CC(C)(CNC(C1CCC(C(C)C)CC1)=O)NC(=O)C(O)CC(N)=O N1(CC(=O)NC2CC(NC(=O)CCC(F)F)C2)C(=O)c2ccccc2C1=O C1(NC(C(C)OCC)=O)CCCN(C(=O)Cc2cc[nH]c2)CCC1 N1(C(C(CC)n2nccc2C)=O)CC=CC(C(=O)N(C)Cc2cc[nH]n2)C1 C=CCCC(=O)NCC(CNC(c1cn(C2CCCC2O)nn1)=O)CO C=CCCC(O)Cc1ccc(C(N2CC(SCC(=O)OC)C(O)C2)=O)cc1 c1(C(=O)OC)c(NC(C2CC3CC3N2Cc2cncc(Cl)c2)=O)cccc1Br Cc1ccc(CCC(=O)NC2CCC2C)o1.C12(CCCC1)C(=O)NCC2 CC1(C)CC(O)(CC(N2CCC(O)(CNC(C3CCC(=O)N3C)=O)C2)=O)CO1 C1(c2c(C)cncc2)NCCC12CNC2 c1(CNC(n2ccc3ccccc23)CC)cccc([N+](=O)[O-])c1 c1(C(=O)NC2C(NC(c3ccn(CCC)n3)=O)CCC2)cc[n+]([O-])cc1 C1(NC(C(CC#C)O)=O)CCCCN(C(=O)CC2CSCCO2)C1 C1(CNC(CNC(=O)NC)=O)CCN(C(=O)CC2CCCC(F)(F)C2)C1(C)C C(=O)(CC(C(F)F)NC(c1ccnnc1O)=O)N1C(CC)CC(C)C1 C1(O)(CNC(C2(C(C)N)CC2)=O)COCCC1O.C1(=O)CNC1=O.C1(C)CC1 CC1CN(C(=O)CCCC2CCC2)CC(C)N(C(c2cc(N)cc(F)c2)=O)C1 N1(C(C2N(CC)CC2)=O)CC2(CCN(C(=O)CCC3CCCCN3C)CC2)C1 c1(C(=O)NCC(C(=O)N(C)CC2(C)CCCO2)OC)cc(CO)oc1C C1(N)CCN(C(=O)CC(C)(C)N(C(=O)CCC2CC(OC)C2)CC)CCO1 C(C)(C)(CC(=O)N1CCOC(C2CC(O)(NC(=O)Cc3ccsc3)C2)C1)N(C)C C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCC1C(NC(COC(C)=O)=O)CCCC1 N1(C(c2ccc(C)cc2)=O)CCC(NC(=O)C(F)CC(C)C)C1(C)C C1(C(=O)NC2CCCN(C(=O)CCc3ccncn3)C2)C(F)(F)C12CCC2 C#Cc1cc(OCc2nc(C(C)C)ns2)ccc1Cl C1(NC(C(C)OCC)=O)CC2CC(NC(=O)CCc3ccccc3)CC12 CN1CCN(C(C23CSCC2C3)=O)CC1C(=O)NC1(CF)CCCC1 C(=O)(C1=NOC2(CCOC2)C1)NCC12C(CN(C(CNC=O)=O)C1)C2 C1(C(=O)Nc2nn[nH]n2)C2CN(C(C3CC4CC4C3)=O)CC12 CCC(C)(CC)C(=O)NCC1CC(NC(C2(C3CC3)CC2)=O)C(O)C1 CCC(CC)C(C)C(=O)N(C)CC1C2CN(C(c3ccc(C(F)(F)F)s3)=O)CC12 N1(C(c2sccc2I)C(=O)Nc2ccc(OC)cc2)CC2CCC1C(O)C2O N1(C(CCC(C)SC)=O)CC(C)CN(C(=O)Cc2c[nH]c(=N)nc2O)CC1C C1(C(N(C(CNC(C=Cc2n(CC)ncc2)=O)C2CC2)C)=O)CCC2(CCC2)C1 N1(C(CCCN(C)CCO)=O)CCC2(CC1)CCN(C(C1CCCN1C)=O)CC2 C1(C)(CC(=O)NCCOCCN(C(=O)C(C2CC2)C2CC2)C)CCCO1 CCCCC(C)(F)C(=O)N1CCC1Cn1cc(CN2CCS(=O)CC2)nn1 CCC(C(=O)NCCC1CC(NC(c2cc(O)nn2C)=O)C1)C(C)(F)F N1(C(CCN(CCC)C)=O)CCC(NC(c2oc(C(C)C)nc2C)=O)C1C c1(C(N2C3C(NC(CC(=O)N(C)C)=O)CC(CC3)C2)=O)nn2cccnc2c1Cl c1(NC(N(C(CNC(N)=O)C2CC2)C)=O)ccccc1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)NC(C(C)OCCc1ccccc1F)=O C1(C)(NC(c2c(C)cco2)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 C12(C(=O)NC3CC(NC(=O)Cn4nc(Cl)ccc4=O)C3)CCOC1CC(=O)NC2 N(C(=NCCF)N1CCC(c2cccnc2)C1)Cc1nc(COC)on1 Cc1cc(C(=O)NC2CCCN(C(C3(CO)CCCCC3)=O)C2)c(Br)cn1 c1(NC)cc(C(N2CC(O)(CNC(c3occc(=O)c3OC)=O)C2)=O)cc(Cl)n1 C1(C(=O)NCC(CNC=O)(C)C)Cc2c[nH]cc2S1(=O)=O.Cc1cc(SC(F)F)on1 c1(CN(CC(CN(C(C(c2ccccc2)C)=O)C)O)C)cc(F)nc(F)c1F c1(C(=O)NCCN(C(C(CC)F)=O)CC2CC2)c(C)oc(C)c1Br c1(C(N(CC(CN(C(C=Cc2c(C)ncs2)=O)C)O)C)=O)[nH]cc2c1CCCC2 N1(C(C2(C#N)CCOCC2)=O)CCC(F)(F)C(NCc2cc3ccoc3cn2)C1 c1(SC(C(=O)N(C(C)CNC(c2csc(-c3ncc[nH]3)n2)=O)C)C)ccccc1 Cn1ccc2cc(C(=O)NCC3CN(C(C4CC4CN(C)C)=O)C3)cnc12 c1(C(N2CC3C(NC(C=CC(C)C)=O)C3C2)=O)ccc(N)cc1S(N)(=O)=O C1(NC(C2C(C)C2)=O)CC2CC1N(C(C1(c3ccc(F)cc3)CCCCC1)=O)C2 c1(CN2CCN(C(=O)NC3CCCN3)CC2)ccc(F)cc1C(F)(F)F c1(NC(C2(CN(C(CC(C=C)c3ccccc3)=O)C)CC2)=O)ccc(N)c(O)c1 c1(C(=O)NC(C(C)NC(=O)CN(C2CCCC2)C)CO)cc2n(c1)CCSC2 N1(C(C(C(CCC)NC(=O)C(C)SC(C)C)O)=O)Cc2cccc(F)c2C1 CC1(CNC(=O)Cc2ccc(CO)cc2)CCCN1C(c1ccsc1Cl)=O Cc1cc(C(=O)NCC(CNC(=O)CC(C)(C)C#N)CO)cc(C)c1F C1(N(C)C(c2ccsc2Cl)=O)CC2CC1N(C(c1cc(O)cc(F)c1)=O)C2 c1(C(=O)NCC2C(NC(c3c(CCC)nco3)=O)CC2)cc2cccc(C)c2[nH]1 C1(CN(C(=O)CNC(c2cccnc2)=O)C(C)C)CCC(C)C1 C1(C(N(CC(C)C(=O)OC(C)(C)C)CC)=O)COCCC12CN(C(=O)C(C)(C)C)C2 N1(C(CCC=CC(C)C)=O)CCC(C(=O)NCCc2ocnc2CO)C1C CC(C)(C)CCCCC(=O)N1CC=C(CCNC(C2CN3CCC2CC3)=O)CC1 C1(C(=O)NC(c2ncc(C(=O)N(CCCN=[N+]=[N-])CCO)s2)C)CCCC12CC2 c1(C(=O)NC2C(NC(C(CC)SC)=O)CC2)ccc(C#N)n1C c1(N2C(C)(C)CC(CO)CCC2)ncnc2c(Br)cccc12 c1(OC)cccc2sc(NC(CN(C)C)CC(C)C)nc12 Cc1ccc(C(=O)NC(C)CCNC(=O)CCc2sccc2Br)cn1 C(=O)(C(C)N=[N+]=[N-])NC1C(CNC(C(COC)C)=O)COC1 c1(C(=O)NCC(CN(C(CC(=C)C)=O)C)C)cnc(OC)nc1COC c1(OC)ccc(-c2cnc(C3CCCN3C(=O)C(O)O)[nH]2)c2cn[nH]c12 N1(C(Cc2cccc(C)c2)=O)CCCN(c2nnc(-c3ccon3)s2)CCC1 Cc1[nH]nc(C(=O)NC2CCC2CNC(c2ccc(CO)c(Cl)c2)=O)c1[N+](=O)[O-] C1(CC(=O)Nc2c(OC)nn(C)c2)CC2(C1)CN(C(c1ccsc1Cl)=O)C2 CCCCCCCCC(=O)N1CCN(C(C2CC3(C2)CC(O)C3)=O)CC(C)C1 c1(OC)n[nH]cc1C(=O)N(CCCNC(C1CCC1C(C)(C)C)=O)C N1(C(c2nc(OC)oc2)=O)CC2CC2(CNC(C2CCOC2)=O)C1 N1(CC(CCC(=O)OC)C(=O)N(C)C)CCn2c(C3CC3)nnc2C1 n1(CCCNC(CN2CC(C)C2)=O)cc(-c2cccnc2)nn1 CS(C)(=O)=Nc1ccccc1C(=O)NC1COCCC1NC(C12CCC(C1)C2)=O c1(CC(=O)N(CC(C)NC(c2ccnc(F)c2F)=O)C)cc(F)cc(F)c1 S(=O)(=O)(c1nc(NC2CCc3c(nnn3C)C2)ccc1Br)NC(C(CC)CC)C C1(CC(=O)NC(CCNC(c2c(CC)n[nH]c2)=O)C)CCCN(CC(F)F)C1 c1(C(=O)NC(C(CO)NC(C(n2ccc(C)n2)C)=O)C)cc2sccc2cn1 c1(C(=O)NCC(CCNC(Cc2cc(C)sc2)=O)O)cc2c(Cl)cccn2n1 C(=O)(CCCCCC(C)C)NCC1N(C(Cc2ccc(OC)nc2)=O)CC1 C1(O)(CCNC(C2COCCO2)=O)CN(C(C2CC2c2ccc(Cl)s2)=O)C1 CC(C)CC(O)C(C)C(=O)NCCCOCCCNC(=O)C(F)(F)CC1CC1 C1(CNC(=O)NC(COC)C)CCC=CN1C(=O)OC.C(=O)(CN(C)C)O N1(C(CSCc2cn(C)nc2)=O)CCCCC(NC(=O)C(F)CC2CC2)CC1 C1(CC)CN(C(c2cnn3c2CCC3)=O)CCN1C(=O)Cc1ccc(C)cc1C C(CNC(C1CC(F)C1)=O)(CC(F)(F)F)NC(c1c(Cl)cc(C)s1)=O C1(C(C(=O)OC)F)CCN(C(c2cnn(C(F)F)c2)=O)C1 C(=O)(C(F)(F)C(O)C(C)C)N.C(=O)(CN(CC(C)C)C)NCCOC C1(C(=O)NC(C)C(C)(C)C#N)CCCCCN1C(=O)CCCN(C)C C1(C2CCCO2)COC(C2CNC2)CN1.N1(C(=O)C)CCC(c2cncnc2)CC1 c1(C2C(NC(C(=O)NC3CN(CC4CC4)C3)=O)C2)ccc(Br)c(Cl)c1 N1(CCC(=O)NC(CCN(C(CC2N(C(C)C)CCC2)=O)C)C)CCNC(=O)C1 C1(C(=O)OC2CC(=O)N(C)C2=O)COc2ccc(F)cc2C1 N1(C(c2c(C)nc(C3CC3)o2)=O)CCCC(C2CC2NC(=O)CNS(N)(=O)=O)C1 Cc1c[nH]c(C(=O)NC(C2CC=CCC2)C(=O)N(CC(C)(C)CO)C)c1C C(=O)(C1=CC(O)C(NC(C2CC(C)(C)C2)=O)C1)NC(COC)C1CC1 C1(C(=O)NC2CCCC2CNC(c2cnc(C3CC3)s2)=O)(CC)CC1(F)F c1(N(C2CCSCC2)C)nc(=N)[nH]c(=NC(CF)C2CCC(C)(C)CC2)[nH]1 C1(c2nnnn2CCC2CC2)(OCC)CCN(CC2CCCN(SCC)C2)C1 Cc1nc2n(n1)CCN(C(C1CC3(CCN1C(c1nnc(S)n1C)=O)CC3)=O)C2 Cc1cc(C(=O)NC2(C)CCN(C(=O)CN3CCC(C)(O)C3)C2)c2n[nH]cc2c1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(N=c2[nH]cnc3cnn(C)c23)CC2(CCC2)C1 C(=O)(CC(C(C)=O)Sc1nnc(-c2cccc(C#N)c2)n1CC(C)C)OCC C1(C(=O)NCC(CC)C)(CCOC)CCN(C(c2ncc(C)cc2C)=O)CC1 C1(NC(C(C)Cc2ccccn2)=O)CCCCC1NC(c1cnco1)=O c1(C(=O)NCCCN(C(C(CC)OCC)=O)C)cc(Cl)c2cc(Cl)ccc2n1 CCC(C)(COC)C(=O)N1CCC(CNC(=O)C(C2CC2)N(C)C)C1 C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(=O)CC2CC=CC2)CC1 C1(C(=O)NC(C(C)C)C(C)NC(=O)C=Cc2ccnn2C)CCC2(CC1)CC2 c1(C)c(C)cccc1Cl.c1(OC)ccc(CNCC2CCCCC2N)cc1 CCN=c1[nH]c(C(N2CCCC(C)(CNC(C3CC(OC)C3)=O)C2)=O)cs1 N1(C(C2(C=C)CC2)=O)CCC2(CC1)CC2NC(c1ncccc1OC(F)F)=O C(=O)(CCC(N)CO)Nc1cc(C(=O)NC)ncc1 Cn1ncc2ncc(-c3nc(CCSC)nn3Cc3ccccc3F)cc12 C(=O)(C(C)(C)CC(C)C)N(CC(CN(C(C(CC(C)C)NC(C)=O)=O)C)O)C CP(C)(=O)C(CO)NC1CC1C(F)(F)F C1(C(=O)NCC2CCN(C(c3cn(C(C)(C)C)nn3)=O)CC2)CCC2(CCC2)C1 CC1(C)CCCCCC1NC(c1ccc(C(F)(F)C(F)(F)F)s1)C1CC1 c1(C(N(C(C(=O)NCc2c(CC)noc2C)C)C2CC2)=O)cncn(C)c1=O C1(NC(C(C)SC(F)(F)F)=O)CN(C(c2ncoc2CN(C)C)=O)CC2CC12 C(C(CC1CC1)C(=O)NCCC1C=CCC1)NC(C1(C)CCC1)=O C1(C(=O)NC(C2(O)CCN(C(C3(O)COC3)=O)C2)C)CCC2(CCC2)CO1 C(=O)(C(CCc1ccsc1)NC(c1c[nH]cc1C(C)C)=O)OC c1(C(=O)NCc2oc(C(N(C(CSC)C)C)=O)c(C)n2)cc(C)nc(O)n1 C1(CNC(c2cc(C)no2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1C c1(C(=O)NCC23C(CN(C(CCCCC#C)=O)C2)C3)sc2[nH]cnc(=O)c2c1C Oc1ncncc1-c1nc(OCC(F)(F)F)nn1-c1cccnc1 N1(C(CCC(C)C)=O)CCN(C(c2cccc(-n3cncn3)n2)=O)CC2(CC2)C1 Cc1cc(CNC(C2CC2C(=O)Nc2ccccc2-c2ncccn2)=O)ccn1 c1(C(N(C2CCCN(C(=O)CC3(O)CCC3)C2)CC)=O)cnn2c(C)cccc12 n1(CCCCCO)ncc(Cl)c1C(=O)OC(C)(C)C.C12CCC(CC1)C(=O)N2 C(=O)(C(CC)C(=O)NCC1CCCN(C(C2CCCCO2)=O)C1)OCC C(C(C)(C)C(=O)Nc1cccc(CNC(=O)C(C)(C)C2CCC2)c1)SC CCCC(CC)C(=O)NN(C(C1(OC)CC(CO)C1)=O)C.C1(F)(C)CCCC1 C#CCC(C(=O)NCC(C1(O)CN(C(c2nnsc2C2CC2)=O)C1)(C)C)C1CC1 C1(C(=O)NC(CC#C)C(=O)NC)C2CC3C(C2NC(C2CC(C)=NO2)=O)C13 N1(C(C(=O)NCCCC)C2CC2Cl)CCOc2c(C(=O)OC)cccc2C1 N1(C(C2N(C(C)=O)CCC2)=O)CCC(NC(c2nnccc2C)=O)C2(CCC2)C1 N1(C(CC(C)(C)C#N)=O)CCCC2CN(C(C34CCN(CC3)CC4)=O)CCC12 c1(C(=O)NCC2(CNC(C(CC)OC3CCC3)=O)CC2)ccc(N=S(C)(C)=O)s1 c1(C(C)OCC(N2CCCC(C(=O)OCC)C2)=O)oc2ccccc2c1Cl CCCCC(CC(=O)NCCC1(O)CCCC1)NC(c1cc(Cl)no1)=O c1(C(=O)NCCNC(C(C(C)C)N(CC)CC)=O)ccc(O)c2c1CCCC2 C1(CC(=O)NC2CCN(C(c3c(CCC)n[nH]c3)=O)C2)(OC)CCCCC1 c1(C2(C(=O)NC)CC2)cccc(NC(=O)Nc2nc(-c3cccc(Cl)n3)cs2)c1 C(C(CCCC)NC(=O)CNC(C1CCOCC1)=O)NC(C1C(=C)CC1)=O C12(OC)CCC(C(N3CCC(CCNC(=O)CC4CC(=O)NC4=O)C3)=O)(CC1)C2 c1(NC(C2C=CC(C(c3cc(N4CCCC4)ncn3)=O)C2)=O)cc(Cl)ccc1Br C1(C(N(C2CCN(C(C3OCCN(CC)C3)=O)C2)CC)=O)CN2CCN1CC2C N1(C(C=CCC)=O)CCCC(N(C2(CCl)CCCC2)C(C)=O)C1.C(=O)(OCC)N C(=O)(C(O)CC(C)(C)C)N1CC(CCCC)N(C(=O)Cn2ncnn2)CC1 N1(C(=O)CC2CCC2)CC(C2CN(C(C3CC34CC(F)(F)C4)=O)C2)C1 N1(CC(=O)NC(CC)CN(C(C2CCS2(=O)=O)=O)CC)CCC(=O)NC1=O C1(c2cn(CCC=C=C)nn2)CN(C(c2cnc(C)cn2)=O)CCO1 N1(C(CCCN(C(C)=O)C)=O)CCCCC1C1CCC1C(=O)NCCN(C)C N1(C(C2(C#N)CC3CC3C2)=O)CC2COCC(C1)C2NC(=O)C(F)=C1CCCC1 C(=O)(C(N=[N+]=[N-])C(C)C)NCCCCCCN(C(C1(CC)CCC1)=O)C c1(C(=O)NC2CC3(CCN(C(=O)CC(O)C4CC4)C3)C2)ccc2c(c1)C(=O)NC2 c1(CNCc2ccc(Sc3cccc(Br)c3)cc2)csc2cncn12 N1(C(CC(CC)OC)=O)CCCC(NC(c2ccc(F)c(Cl)n2)=O)CC1 C1(NC(=O)Cc2csc(C(F)(F)F)n2)CS(=O)(=O)CC1NC(c1cc(Br)n[nH]1)=O CC1CCCN(C(=O)C(C)(CO)NC(C2CN3CCN2CC3)=O)CC1 Cc1nc2c([nH]1)CC(NC(C1CCCN1C(=O)C(C)N(CCO)CCO)=O)CC2 CCC(O)C(F)(F)C(=O)N1CC(NC(c2cnc(C3CCC3)nc2O)=O)C1 C1(C(N2CCC(C)(CNC(c3c(C)noc3N)=O)C2)=O)OCCN(C)C1=O c1(C(=O)NC2CCCN(C(C(CC(=C)C)OC)=O)C2)ccc2nonc2c1 c1(C(N(CC(C)CNC(=O)C(=O)NCC2CC2)C)=O)cn2c(n1)CCC2 c1(C(=O)NC2CC(C(C)NC(Cn3ncc(CC)c3)=O)C2)n[nH]cc1[N+](=O)[O-] c1(C(N(CC(C)N(C)C(c2ccc(N)cn2)=O)C)=O)cccn2nccc12 C1(CNC(C2(C)CCCOC2)=O)CN(C(=O)CCOC2CCC2)C2(CCC2)C1 c1(C(=O)NCC(N(C)C(C2C3CC4C(C3=O)C24)=O)C2CC2)ccc2cnnn2c1 N1(C(=O)C=CCc2ccccc2)CC2(C1)CN(C(C1(c3cccc(F)c3)CC1)=O)C2 c1(C(=O)NCCCCNC(c2cc(CCOC)on2)=O)cc(F)cc(F)c1F Cc1nn(C)cc1-c1ccc(NC(c2cc(Cl)ccn2)=O)cn1 Cc1cc(C)c(C(=O)NC2CC(CNC(=O)CCn3ncn(C)c3=O)C2)cc1C C1(CNc2ccn(C3CNC3)n2)CC12CN(C(=O)NC(=O)OC)C2 N1(C(C2C(OCC)C2)=O)CCC(C2(NC(C3CN(C(=O)NC)C3)=O)CC2)C1 Cc1cc(C(=O)NCC2CCCN2C(c2ccn3c2CCC3)=O)nc(Cl)c1 C1(C(C)(C)C)CN(C(C2CC2C2CC2)=O)CCN1C(=O)Cc1csc(Cl)n1 C1(C(=O)NC(C(CO)NC(c2nc(C)sc2)=O)C)CCC(C)(C)OC1 c1(C(C(N2C(CNC(CC=CCC)=O)C(C)CC2)=O)=O)sc2ccccc2c1C N1(C(CN(C(=O)CN2CCC(OC)C2)CC#C)=O)CCC2(CCOC2)CC1 Cn1ncc2c1CC(C(=O)NCC1CN(C(c3ccncn3)=O)CCCO1)CC2 N1(C(CCc2c(C)n(C)nc2)=O)CCN(C(c2cncc(C(N)=O)c2)=O)C(C)C1 c1(C(=O)NCc2ccc(C(N3CC(C4CCCO4)C3)=O)s2)ccccc1C1CC1 c1(C(=O)NCC2(CNC(Cc3cc(C)n(C)n3)=O)CC2)cc(O)cc(=O)o1 Cc1ccc(C=CC(=O)NC23CCC(NC(C4CC5CCC5C4)=O)(CC2)C3)c(C)c1 CC1(C)CC(CNC(c2scnc2Br)=O)N(C(=O)CN2CCCC2=O)C1 CCC(Cc1cn(CC(=O)Nc2ccccn2)nn1)C(=O)NC1CCCO1 N1(C(C=NOC)=O)CCN(C(c2cc3c(s2)CCC3)=O)C(C(F)F)C1 Cc1nc2ccccn2c1CN1CCNC(CO)C1 N1(C(c2n(C)nc(O)c2)=O)CCN(C(C23OCC(OC(C)(C)C)(C2)C3)=O)C2CC12 N1(C(C2CCN(C)CC2)=O)CC=C(C(C)(C)C(=O)NCc2nn(C)cc2CO)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CCCN(C(=O)Cn2cncn2)CC1 c1(CC(=O)NC2CCC(Cn3cc(CC4CCC(=O)C4)nn3)C2)cc(F)ccc1Cl C(=O)(CC(C(C)C)NC(C1(CCC)CC1)=O)NC(C=C)C(F)(F)F CCC(CNC(C1C(CN=[N+]=[N-])C1(C)C)=O)(CC)NC(=O)C(C1CCC1)OC c1(C(=O)NCC2CC(F)(CNC(C3CCN(C)C3=O)=O)C2)cccc2sncc12 C1(CNC(CS(CC)(=O)=O)=O)CC2OCCC2N1C(c1ccc(C)c(C)c1)=O N1(C(C(C(CC)C)NC(C2CC(SC)C2)=O)=O)CCCC2CC1C2(C)C c1(C(=O)OC)nc(=NCC2(C)CCCN(C(=O)C(F)OC)C2)c2c([nH]1)CCC2 C12(CC(=O)NCC(=O)NC(C)(C)C)CCC1CN(C(c1c[nH]c(=N)o1)=O)C2 N1(C(CC2CCC(C)C2)=O)CCC2(CC1)C(NC(=O)CC1CN(C)C1)CS2(=O)=O Cn1c(CCC(=O)NC(CC2CC2)C(=O)NC(c2ccccc2)CO)nnc1S c1(CC)cn(C)nc1C(=O)NCC1CC1CNC(=O)C=Cc1cocn1 C1(CC)CCN(S(=O)(=O)N2CCC(c3nc(=N)n(C)[nH]3)CC2)CC1COC c1(C(=O)NCC2CC(NC(CC3C(C)OCC3)=O)C2)ccc2oncc2c1 c1(C(=O)NCCOC2CCN(C(C3C(C)C3)=O)C2)c(O)ccc(Br)c1Cl C1(CNC(CCc2cc(C)[nH]n2)=O)CC(NC(=O)C=Cc2scnc2C)C1(C)C c1(OCC)ccccc1C(=O)NC(C)(C)CCCNC(=O)CC(CC)OC c1(C(N2C3CC(NC(C(C)NS(C)(=O)=O)=O)(C3)C2)=O)ccc(F)c(S(C)(=O)=O)c1 c1(C(=O)NC(CNC(C(CC=CC)C)=O)COC)ccc(O)cc1C C1(C(N)=O)CCC(CNC(=O)CC2CC(NC(C3CC4(CC4)C3)=O)C2)O1 N1(C(C(C)SC)=O)CCCCCC(NC(c2sc(OC(F)F)nc2C)=O)C1 C#Cc1ccnc(C(N2CCC(NC(=O)CCOC(C)C)CC2C)=O)c1 C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCCc2cnccn2)C1)OC c1(C(=O)NC2C(NC(c3c(C(F)(F)F)nc(C)s3)=O)C2)ccnc2c1CCC2 c1(CN(CCC(C)(C)C#N)C2CC3CNC2C3)c(Cl)c[nH]c2nccc1-2 C(=O)(C1=C(Cl)CCOC1)NCC12N(C(CCOCCN(C)C)=O)C(CC1)CC2 N1(CC)CCC(NC(=O)CCCn2cc(C3CCCC3)nn2)C(C)C1 c1(NCCN2CCN(Cc3cn(CC(CC)O)nn3)CC2)cc2[nH]ccc2s1 C(=O)(C(F)(F)CC1CC1)NC(C1CCN(C(=O)CC2C=NN(C)C2=O)CC1)C C#CCCCCC(=O)NCC1(OC)CN(C(=O)CSC(F)(F)F)C1 C1(CNC(CCC2CCC(NC(C3(CC)CC3)=O)C2)=O)CCC(C)(C)CO1 c1(NC)ccc(F)c(NC(C2OCCC2CNC(=O)CCN2CCOC2=O)=O)c1 C1(CNC(Cc2cc(C)sc2)=O)(NC(c2ccc(C#N)s2)=O)CCCCC1C CC1CN(C(C2(C)CCCN2C)=O)CC(C)N1C(=O)CC1CCCCCCC1 S(=O)(=O)(c1cnc(NCCn2cnnn2)c(Cl)c1)NC1(CO)CCCC(C)C1 N1(C(COCC)=O)CCOCC(CNC(=O)CCc2ccc(Cl)c(F)c2)C1 Cc1ccc(NC(=O)C(=O)Nc2cccc(N3CCCCC3)c2)c(C)c1 C12(C(N3CCC(N(CCC)C(c4coc(N(C)C)n4)=O)C3)=O)CCC(OC)C1C2 c1(CC(=O)N(C)CCOCCN(C)C(C2CC2c2ccco2)=O)cccnc1Br Cc1csc2ncc(C(=O)NC(C)C(C)(C)NC(=O)C(C)(F)F)c(=O)n12 N1(C(c2n(C(C)C)ccc2)=O)CC(CCNC(C2CCCO2)=O)C(C)C1 CC1(C)CC(NC(c2ccoc2)=O)CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 C1(CC(=O)NC(C2CCOCC2)C)CCCN(C(C2(C)CCN(C)C2)=O)C1 c1(CC(=O)NC(CN(C(C(CC)OC)=O)CC)C)sc(C)nc1C Cn1cncc1C(=O)N(CCNC(c1csc(-c2cccs2)n1)=O)CC1CC1 Cc1noc(C)c1CCC(=O)NCC1COCCN1C(C1CCCC1(F)F)=O Cn1ncc(C(=O)NC2CN(C(C3(CF)CC3)=O)CC3(CC3)C2)c1S(C)(=O)=O c1(C(N(CC(CNC(C2(COC(C)C)CC2)=O)(C)C)C)=O)ccn2nccc2n1 C1(NC(c2c(C)ocn2)=O)C(C)(C)C(NC(=O)C(O)CC2CCCCC2)C1(C)C c1(OCCOC)ccc(C(=O)N(C(C)CCNC(=O)CCC=C(C)C)C)cn1 C(C1=CCN(C(c2ccccc2-n2ccc(C)n2)=O)CC1)NC(CSCC=C)=O C1(NC(C(CCC)O)=O)COC2C(NC(=O)C=CSc3nc[nH]n3)COC12 C(c1ccccc1C(F)(F)F)=CC(=O)NC(CSC)C(=O)N(C)CCO C1(NC(C(CC#C)NC(c2nn(C)cc2C)=O)=O)CC(C)N(C)CC1C C(=O)(C1Cc2ccc(Cl)cc21)NC(C(C)NC(=O)CCCCN(C)C)CO C#CC1(C(=O)NC2CCC(C3CC3)C2)CCN(C(c2cnc(N(C)C)nc2)=O)C1 Cc1cc(C(=O)NCC(CNC(=O)CCc2ccccn2)CO)nc(O)n1 C1(C(=O)Nc2c(OC)cc(F)cc2)CN(C(C2CC2C2CC2)=O)CC(F)(F)C1 CC1(C)CCOC1C(=O)NCC(C1CCOC1)NC(=O)CN1CC(=O)NC1=O C1(NC(C(C)C2CC2)=O)Cc2ccccc2C1NC(c1cnsn1)=O C1(=O)CCC(N(C)C)C(=O)N(CC)CC(=O)O1.n1(CCNC(C)=O)cc(C)cn1 c1(C(N(CC(=O)O)Cc2ccccn2)=O)cccc(SCc2n[nH]cc2Br)c1 n1(C(C)C)cnc(C(=O)NC2CC(C(F)C(=O)NC(CN3CCCC3)CO)C2)n1 c1(OC)cc(-n2nnnc2C(CCC(F)(F)F)Nc2ccccc2C)ccc1F C1(C(C)C)(C(=O)NC(C)(C)CCCF)CCCN1C(=O)C(Cl)Cl C(=O)(CC1=NNC(=O)C1)NCC1CN(C(c2nc(CC)oc2)=O)C(C)CC1 C=CC1(CC(=O)NCC2CCN2C(c2cscn2)=O)CCC1 c1(C(=O)NC2C(CNC(c3ccc(C(N)=O)[nH]3)=O)CC2)[nH]cc2c1CCCC2 c1(C(C)(C)C)ccc2oc(CN(C(N)=O)CC3CC34CCOC4)cc2c1 N1(C(C(CCC)NC(N)=O)=O)CCC=C(C(=O)NC(C)C)C1.C12CC(C1)N2 CC(C)(C)CC(O)CC(=O)N1CCC1c1cccc(OC(F)(F)F)c1 C1(C(N2CCC(NC(CS(=O)(=O)N(C)C)=O)CC2)=O)CN2CCCCC2CO1 C1(C(N(C2CC(C)C2)C)=O)C2CCC(C2)N1C(=O)CC(O)C1CCCC1 c1(C(=O)NCCC(C(C)C)NC(C(C(=C)Cl)(C)C)=O)ccc(S(=O)CC#N)cc1 C(=O)(C(Cc1ccccc1)S(C)(=O)=O)N1CCC(NC(C2(OC)CCC2)=O)CC1 C1(CC(=O)NC23CC(C(=O)NC(c4nnn(C)c4CO)C)(C2)C3)CC2CCC1C2 C12(NC(CSCC(C)C)=O)CCN(C(=O)Cc3ccccc3C#N)CC1C2 N1(C(C(c2cccc(Cl)c2)OC)=O)CCC(C2CCN(C(=O)C=C(C)C)C2)C1 N(C)(C1CN(C(c2ncc(CN)s2)=O)CCc2ccccc21)C(COC(C)(C)C)=O CC(O)CCCC(=O)NC(C)CCNC(=O)C1=NNC(=O)C1 C(=O)(CCCCCN=[N+]=[N-])N1CCCC(CC(=O)N(C2CCC(O)CC2)C)C1 Cn1cc(C(CO)NC(=O)CC2(C)CCN2C(=O)C=CC(=O)N(C)C)nn1 Cc1cc(NC2(CO)CCCN(C(=O)CC(C)C(F)(F)F)C2)ccc1[N+](=O)[O-] c1(C(=O)NCC2CCN2C(=O)Cc2ccc(Br)cn2)nc2ccccc2s1 C=C(Cl)CC(C(=O)N(CCN=[N+]=[N-])C)NC(=O)CCNC(N)=O c1(CNC(C(=O)NC2CC(SC)C2)=O)ncc(C(C)(C)C)o1 Cn1ncc2c(N3CC4(CC4)CC3CNC(C3(C(F)F)CC3)=O)ncnc12 c1(OCC)cc(C(=O)NC2CC(CNC(c3sccc3OC(C)C)=O)C2)ccn1 c1(C(=O)NCc2cccc(NC(C3C(C)COCC3)=O)c2)ccc(F)c(N)c1 c1(CN(CCNC(C2CC2(c2ccccc2)C)=O)CC)nc2cnccc2[nH]1 N1(C(C(C)N(C(C)C)C2CC2)=O)CCC(NC(=O)CCc2ccccc2Cl)CC1 N1(C(C2C(C)(CC)C2)=O)CC(O)(C2(CNC(=O)CN(C)CC)CC2)C1 C1(NC(C(COC)(C)C)=O)CN(C(=O)C=CCOC2CCOCC2)C(C)(COC)C1 N1(C(=O)NCCn2cnc(=N)[nH]2)CCS(=O)(=O)C2(CC(C(=O)ON)C2)C1 O=C(C1CCOc2ccc(F)cc21)NCC1CCCCN(C(C2CCC2)=O)C1 n1(CC)nc(C(N2CCC(C(C)NC(=O)CC(CC)C3CC3)CC2)=O)cc1C CC1CN(C(C2CCC2C)=O)CCCN1C(c1ccc(-n2ccnn2)cc1)=O O=C(CC1OCc2ncccc21)NC1CN(C(c2cccc(O)n2)=O)CCC1F CC1CCCn2ncc(C(=O)NC3CCCCN(C(=O)CCc4cscn4)C3)c21 N1(C(c2c(C)ccs2)=O)CCC2(CC(C(=O)N3CCCCC(C)(C)C3)=NO2)C1 C(=O)(C(C)(C)CNC(c1nccnc1CC)=O)N1CCC(N(C)CC)C1 N1(C(Cc2ncn(C)c2)=O)CCCCC1CCNC(=O)CCC1CCCOC1 Cn1cc(C2=NOC(C(N3CC4CCN(C(c5cnsc5)=O)CC4C3)=O)C2)cn1 Cc1ccc(CNc2ncccn2)c(Br)c1 c1(C(N)=O)cccc(F)c1C(=O)NCC1(NC(=O)C(c2ccccc2)O)CCC1 N1(C(C(COC)NC(C)=O)=O)CCC(NC(c2cc(SC(C)C)nn2C)=O)CC1 C1(C(N2CCCC(=C)C2)=O)CC2OCCC2N(C(c2ccc(O)cc2)=O)C1 Cc1ccc(C(=O)NC(C)CCCNC(C2CC2c2cnc[nH]2)=O)c(N)c1 Cc1cc(CC(N2CC(NC(c3cnc(O)cc3O)=O)CC(O)C2)=O)cc(F)c1 C1(N(C(C(C)OCCC=C)=O)CC)CCCN(C(c2ccnn(C)c2=O)=O)CC1 N1(C(C2C3CC(NC(c4ccnnc4O)=O)C(C3)C2)=O)CCc2nnnn2CC1 C(CC(=O)NC(C(=O)N(CC(O)COC)C)c1cccs1)OCC C(CC(F)F)(C(=O)NCC1(O)CSC1)NC(c1nc(CCC)oc1)=O C1(C(N2CC(OC)(CNC(c3occc3CN(C)C)=O)C2)=O)CCCN1C=O c1(C(=O)NC2(C(=O)NCC(C(C)C)CO)CCCCC2)cc2ccccc2o1 O(NC(=O)CS(=O)CC)C(c1nnc(C(CCCC)C)o1)c1ccccc1 c1(C(=O)NCc2c(C(=O)NC34C(C)OC(CC3)C4)n[nH]c2)ccn2cncc2c1 c1(C(=O)NC2CCN(C(CC3C(C)C3)=O)CC2O)cc(O)ccc1[N+](=O)[O-] n1(CC)cnc(C(=O)NCC(C(=O)N(CC(C)SC)C)N(C)C)c1 C1(O)(C(C)NC(c2ccc(SC)s2)=O)CCN(C(=O)C=CC(C)(C)SC)CC1 c1(NC(CC2C(NC(=O)OC(C)(C)C)CC2)=O)cccn(C(C)(C)C)c1=O N1(C(C2N(C(=O)OC)CCC2)=O)CC2CC(N3CCCC(C)(O)C3)C1C2 c1(OCCNC(c2cc(Br)c(Br)o2)=O)ccc(C2CCCCC2)cn1 c1(CC(=O)NC2CCN(C(C(C)NC(C)=O)=O)CC2)ccc(C(=O)O)c(C#N)c1 CCCC(C)CC(=O)NCC1(F)CCN(C(c2cc(C3CC3)on2)=O)C1 C1(C(=O)NC2CC3CN(C(C(COC)(C)C)=O)C2C3)Cc2cc(F)cc(F)c2O1 C1(NC(c2c(OC)scc2)=O)C2CCN(C(=O)C=Cc3nc(C)cs3)CC12 C1(C(=O)NCC(C)(O)CNC(C2COCOC2)=O)CCOC2(CCCC2)C1 c1(-c2cc(NC(c3cnc(OC)c(C)c3)=O)ncc2)cccc(C#N)c1F c1(OCCCOC(CS(N)(=O)=O)=O)cc([N+](=O)[O-])ccc1OC(F)F C1(C2CCC2)(C(=O)NC2CN(C(C(c3cn(CC)nc3)=O)=O)C(C)C2)CC1(F)F c1(C(=O)NC(C(C)NC(c2ncncc2F)=O)(C)C)cccc(=O)n1C C1(NC(c2nc(-c3cc(Br)ccc3F)cs2)=O)CCC(F)(F)CC1 N1(C(=O)OC(C)(C)C)CC(NC(=O)NC(=O)CCC(N)=O)C(C(F)F)C1 c1(NCC(N(C(c2c(C)scn2)=O)C)C2CC2)nc2c(cc1C#N)CCCC2 CC1CCN(C(=O)CNS(=O)(=O)N(C)C)C1CNC(=O)CCC=CBr Cc1nnc2n1CC(C(=O)NC(C1CCN(C(=O)C3=NNC(=O)CC3)C1)C)CC2 C1(C(N(CCC(N2CCC(C)(N(C)CC)C2)=O)C(C)C)=O)CC2(CCO1)CC2 Cc1ccc(C(=O)NC2CCCN(C(=O)NC3CC3)C2)nc1 C1(NC(C(C)OCCCC)=O)CN(C(C2(C(F)F)CCOCC2)=O)CC1(C)C C1(CC(=O)NCCCOC=C)CN(C(C2CC2F)=O)C(C)(C)C1 C(CC(=O)NC1C(C)(C)C(NC(C2(C)COC2)=O)C1(C)C)(C(F)(F)F)OC C1(C(=O)NCC(CNC(c2cc(CC)[nH]n2)=O)C)(CC2CCCO2)CCOCC1 c1(COC)ccccc1C1=CCN(C(c2cccnc2C(F)(F)F)=O)CC1 C(=O)(C(C)C1=CCCC1)N1C(CCNC(c2ccc(CC)cn2)=O)CC(OC)C1 c1(C(N2CCC(C(=O)NCCCc3ccccc3Cl)C2)=O)n[nH]c2c1CCC2 C(CCC(=O)NCC1CC1CNC(=O)CCc1cnn[nH]1)SC c1(OC)cc(C=CC(=O)N(C(C)CNC(c2cncc(SC)n2)=O)C)ccc1O c1(C(=O)NC(C)CNC(=O)Cc2cc(OC(F)F)no2)ncc(Br)cn1 N1(C(C(CC)C)=O)CC2CCCC2(CNC(C2(CO)CCC2)=O)C1 CC1CCCCC1(C(F)(F)F)NC(=O)CC1COC(C)(C)C1 Cc1nc2ncccn2c1CN(C1CCC1)C(N1CC(c2ccccc2)C1)=O n1(CC)nnc(C)c1C(=O)NCCCCC(C)NC(=O)CCC1CCC(O)CC1 C1(CNC(c2nc(C(C)=O)sc2)=O)CN(Cc2cc(C)on2)CCCO1 c1(C(=O)NCC(CC)NC(C2(C)CC(C)=NO2)=O)cc(C(F)(F)F)ccc1OC c1(C(=O)NCC2C(NC(c3cc(C)sc3)=O)C2)ccc(N2CCCC2=O)cc1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(CC)CC(=O)N1CCCC1CN(C)C C(=O)(C1CCc2nccn21)N1CC(NC(c2c(S(C)(=O)=O)scc2)=O)C1 C#Cc1cccc(C(=O)NC2(CNC(c3ccsn3)=O)CCC(C)(C)CC2)c1F C(=O)(C(CCNC(=O)OC(C)(C)C)CC(C)C)NC(CC)CNC(=O)NC c1(C(=O)NC(CC)CNC(C2CCC3CC3CC2)=O)cc2sc(C)cc2s1 CC(F)(C(=O)N1CCC(NC(=O)CCCSCC(N)=O)C(CO)CC1)C(F)(F)F N1(C(C2(CC=C)CCOC2)=O)CC(C(=O)Nc2c(C)noc2C2CC2)C(SC)C1 C(=O)(C(C#N)C(C)(C)C)NCc1occ(C(N2CCC(C(C)(C)C)C2)=O)n1 Cc1cccc(C(=O)NC2CCCN(C(=O)COc3ccc(F)c(Cl)c3)C2)c1F C=CC1CN(C(=O)COCC2CCOC2)CC1NC(=O)CNC(=O)CCC(C)C C1(C(N2C(C)CSCC2)=O)CC2(CCC2)CN1C(=O)CC1CC(F)(F)C1 N#CCCCC(=O)N1CCOCC1CCNC(C1(c2ccncc2Cl)CC1)=O c1(CC)ccc(C(=O)NC(CN(C(=O)C(C)N(C)C)C)CC)cc1CC C#CC1CC(NC(=O)C(C)(C2CCC2)NC(=O)CSCCC)C1 Cc1ccc(C#N)cc1C(=O)NCC(C)C(=O)NCC1CN(C2CC2)C1 C(=O)(CN=c1cc[nH]cc1)N1CCCC(N(C)C(c2cc(C#N)ccc2O)=O)C1 C1(NC(=O)CC2CCC2)C2CCC(C2)C1C(=O)NC1C=CCC1 CCC(CC)(CC)C(C(=O)N1CSCC1C(=O)OC)NC(=O)OC c1(C(C)=O)cccc(C2CCC2)c1.c12ccc([nH]1)C(=O)N1CC(C1)N(C)C2=O N1(C(c2cc(C)ccc2OC)=O)CCC(C(=O)NCC2CC(CF)C2)C(C)(C)C1 N1(C(C2(C)CCOC2)=O)CCOC2(CCC(NC(=O)Cc3ncc(Cl)s3)CC2)C1 N1(C(C=CCN(CC#C)C)=O)CCSCC1CCNC(C1CCCCC1C)=O Cc1ccc(-c2nc(C(=O)NC(C)(C)CCNC(=O)CC(F)F)cs2)s1 Cc1cnc(N2CC(F)(F)CC2CNC(=O)CCOC(F)F)nc1C C(=O)(C1CCCc2ccccc21)N1C(C(C)(C)C)CN(C(=O)CCC(F)F)CC1 c1(COC)ncc[nH]c1=NC1CCCCC1NC(=O)C(F)=C(C)C1CC1 c1(C(N(C(CNC(C(CC=C)C)=O)C)C)=O)c(F)cccc1Br C(=O)(CC(C(C)OC)NC(c1c[nH]c(=O)cn1)=O)N1CCN(C(CC)C)CC1 CC1CC2(CCN(C(C3(CO)CC3)=O)CC2)CN1C(C1CCC(C(F)F)CC1)=O CC1(C)CC(NC(C2CCC(=C(F)F)CC2)=O)CN(C(C2CCCC23CC3)=O)C1 N1(C(C(C)N(C(C(C)C)=O)C)=O)CCCCC1C c1(CC(=O)OCC)ccc(-c2nc(Cc3ccccc3F)nn2CC(F)F)cc1 C1(C(=O)NCc2ccc(N(C)C)c(F)c2)CCOCC12CCCC2 C1(C(=O)NC2(CF)CCN(C(C(C(C)C)F)=O)C2)CC2CCCC(C1)C2 C1(CNCc2c(C)c(C(=O)O)n[nH]2)CC2C=CC1CCC2 CC12CCC(=O)N1CCCN2C(=O)C(c1cccnc1)O C(C(C(=O)NC(C12CC(CO1)C2)C)C(C)(C)C)NC(c1cc(C)ncc1)=O c1(CN=C(NCCOC)NC2CC2C)ccc(C#N)c(F)c1 C1(CNC(CCN(CCCCC)C)=O)CN(C(=O)C(OC)OC)CC12CC2 N1(C(c2cc(C(=O)OC)[nH]c2)=O)CC2CCCC2(CNC(=O)CN(C)C(C)C)C1 C1(NC(c2c(C)cccc2C)=O)CN(C(=O)C(C2CCOCC2)=O)CC(F)(F)C1 c1(C(=O)NCC(C)N(C(=O)COC2CCC2)CC)c(O)nnc2c1CCCC2 Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1NC1CN(C(c2cncc(Cl)c2)=O)C1 c1(CN(C(C2CCN(CCC)C2)=O)C)nn(C)cc1Br C#CCCCCCC(=O)N(C)CC1(C)CCCC1NC(c1scnc1CC)=O C1(COC)CN(C(=O)C(c2ccccc2)OC(C)C)CCN1C(=O)COC C(CO)(CC(F)(F)F)NC(=O)Cc1ccc(Cl)cc1 C1(CNC(=O)C(C)OC)CCCCC1C(N1CC(c2ocnc2CC)C1)=O c1(OC)ccccc1OCC(=O)NC1(CCNC(=O)CC(C)C2CCCO2)CC1 c1(C(N2CC(OC)C(C)C2)=O)cc(C(C)(C)C)nc(Cl)c1 c1(C(=O)NCC2OCCN(C(=O)NC3CC4C=CC3C4)C2)cc(Br)ccc1I c1(NC(C#CC)=O)ccc(C(N2CCCC2c2ccncc2)=O)nc1 N1(C(C(C)OCC#C)=O)CC(F)(F)CC1C(N1CCC(OC(C)C)C1)=O CC(CCC(C)(C)C)NC(=NCc1ccn(CCF)n1)NCc1ccccc1Br c1(C(N2CC3C(CNC(c4c(C(C)C)onc4)=O)C3C2)=O)n[nH]c2c1CCCC2 C12(NC(CNC(C)=O)=O)CCCC1N(C(=O)CC1CC3CCC1C3)CC2 N1(C(Cn2cc(CNC(=O)CCCF)nn2)=O)CCS(=O)(=O)CC1 CC(O)(CC(=O)NCCC1(O)CN(C(C2CC3(CCC3)C2)=O)C1)C1CC1 CC1CC(CNC(=O)Cc2ccc(C3CC3)cc2)CN1C(c1nonc1N)=O N1(C(c2cc(OC)n[nH]2)=O)CCC(NC(=O)COC2CCCCC2)C(O)C1 c1(C(N(CCC(=O)NCC2CCN(CC)C2)C2CC2)=O)ccc(C)cc1 c1(C(N2CCC(NC(CCC(=C)C)=O)(CC)CC2)=O)cc2cccnc2nc1C C(C(CC(C)C)NC(=O)C(O)CC1CCCC1)NC(CC1(CC(=O)OC)CC1)=O c1(C(=O)NC2CC(n3cc(-c4ccc(N)cn4)nn3)C2)ccc2nn[nH]c2n1 C1(CNC(C(C(C)(C)O)F)=O)C2CCCC1N(C(c1cc3sccc3[nH]1)=O)C2 C1(CC)CCCN(C(=O)CC(COC)NC(=O)Cc2cccnc2O)C1 N1(C(c2c(C)onc2-c2ccccc2)=O)CC2CN(C(C3(C)CC3F)=O)CC2C1 c1(CN2CC(CNC(c3ccc(C)s3)=O)OCC2)c[nH]c2cnccc12 c1(C(=O)OCC(C)=O)ccn2ncc(Cl)c2n1 CCCCC(=O)C(=O)N(CC(CC)NC(C1CCOC(C(C)C)C1)=O)C N1(C(c2ccn(CC)c2C)=O)CCC2(CCCCN(C(=O)CC3CN(C)C3)C2)C1 C1(NC(C2(CC#C)CCCO2)=O)CN(c2nnc(CO)s2)C2(CCOCC2)C1 c1(OC)cc(-n2nc(-c3cc[nH]n3)nc2CCn2c(C)csc2=O)ccc1Cl Cc1cccc(F)c1CC(=O)NC1CC(CNC(=O)CC(O)C(C)C)C1 c1(COC)nc(NCc2cc(Br)ccc2C)cc(=NCCC2CCCN(C)C2)[nH]1 c1(C(=O)NC(CN(C(c2ccc(OC(C)C)cc2)=O)C)C)cccc(S(C)=O)c1 N12CCN(C)C(C1)C2=O.c1(C(=O)NCC2(CO)CC(=C)C2)ccc(OC)nc1 N1(C(C=C(CC)CC)=O)CC2CC(CNC(c3ccc4occc4c3)=O)CC1C2 N1(C(C2C(=C)C2)=O)CC(C)(C)C(NC(=O)CCSCCCC)C(C)(C)C1 S(=O)(=O)(c1cccc(-c2ccc(Cl)s2)n1)NC1C(OC)CN(C)C1 Cc1ccc2[nH]c(C(=O)NCC(C)CNC(C34COC(CCO3)C4)=O)cc2c1 c1(CC(=O)O)cn(CC2CCC(C(=O)O)C2)nn1 c1(NC(=O)NCCOCCOCCCC)cnn2c(C)ccnc12 C1(CC(=O)N(C2CCCC2)CCOC)CCCN(C(C2CCC=CCC2)=O)CC1 C12(C(=O)Nc3cc(C)c(NC(=O)C(O)C(C)C)cc3)CCC(CC1)C2(C)C CN1CC2CCC(C1)N(C(C1(C)CCN(C(=O)Nc3ccccc3)C1)=O)C2 c1(C(C)NC(=O)C(C2CN(C(=O)CCCF)CCO2)CC2CC2)ccc(F)cc1 C1(C(N(CCCOCCCNC(C2CC2(C)C(F)F)=O)C)=O)CC2(CSC2)C1 N1(C(C2C(C)OCCO2)=O)CCCC12CCCN(C(C1(C)CCN(C)CC1)=O)C2 C1(C(=O)NC2CC(C)(NC(=O)Cc3ccnnc3O)C2)CC1C1CCCC1 CC1COC2(C1)CN(C(C1CC=CCC1NC(C1(C3CC3)CC(=O)C1)=O)=O)C2 n1(CCCC(=O)NCCC2CC2NCC2CCCC(=O)N2)nnc2ccccc12 N1(C(CCNC(C(=CC2CCCC2)C)=O)=O)CCCC(C)C1C(N)=O C1(NC(CCOCCC)=O)CN(C(=O)C=CCSC(C)(C)C)CCC1F C12(C(=O)NC(C(=O)OC)C3CC3)C(NC(=O)C(C)N3CCCC3)C3CC1C2C3 N12CCC(CC1C(F)(F)F)C2.O=C(CCCn1cc(C2CCCCC2)nn1)OC C1(CN(c2nnc(CC)o2)CC)CCCN(C(=O)CSc2cnn(C)c2)C1 C1(NC(=O)Cn2cccn2)CCCC(NC(=O)Cc2c(O)ncnc2O)CC1 N(C(=NCCNC(c1ccco1)=O)NC1CCN(C(=O)NC)CC1)C(C=C)C C(CCCCC(=O)N1CC(N(C)C)C1)N(C(c1cccc(NC)n1)=O)C c1(CC)nc(C(=O)NCC(C)NC(=O)C(C)C2CCOC2)co1 C12(NC(c3ccn(C(C)C)n3)=O)CC1CN(C(=O)Cc1ccc(Cl)cc1)C2 c1(C(C(=O)O)=O)ccc(Cl)c(F)c1.c1(CC)ccnn1C.N1(CC)CCOC1=O Cc1cnc(Cl)c(NC(C2CSCCN2C(c2noc(C)c2C)=O)=O)c1 CC1C(NC(=O)CC2CCC(=O)NC2)CCCN1C(c1ccc(C(N)=O)cn1)=O c1(C(C)=O)ccc([N+](=O)[O-])cc1C(=O)NC1CCCC1NC(C1CC(F)(F)C1)=O C1(OC2(C)CCC2)CCOCC1C(N1CCC(CO)(CO)C1)=O.C1C(=O)N1 C(=O)(C(C(C)C)SC)NC1CC(O)C1.C1(N2C(=O)COCC2=O)CCCC1.CO CCCCCCCCCC(C)(C)C(=O)NCCCN(C)C(C1CCC1F)=O c1(C(=O)NCCNC(C(C2CCCCC2)C)=O)cn(C)nc1C(c1ccco1)=O C(=O)(CCCCCCCBr)NCCNC(C1CC(=O)NCC1)=O Nc1cc(C(N2CCC(NC(C3CC=CCO3)=O)C2)=O)ccc1-n1cnnc1 C1(NC(C(CSC)OC)=O)(CNC(c2csc(C)c2)=O)CC2CCC1CC2 CCC(CC)C(O)CNC(=O)C1=CCC(NC(C2CC(O)C2)=O)C1 N1(C(CC(C)O)=O)CC23CCCC2(C1)CN(C(=O)C=Cc1ccncn1)C3 C1(COC)CC(CO)N(C(=O)CC)C1.c1(C(=O)OC(=O)CO)cnc(C2CC2)nc1 c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cn(C3CC3)cn2)=O)C1)=O Cc1cc(C(=O)NCC2CCCN(C(=O)CCc3ccccc3)C2)cc(C)c1F N1(C(C=CCCC)=O)CCC2(C=C(C(=O)NCC3CCCC34CCC4)C2)C1 Nc1ccc(C(=O)NC2(C(=O)NCC3CCCCC3)CC(F)C2)nc1F C1(C(N(C2CCCC2)CCNC(C2(C)CC2(Cl)Cl)=O)=O)CCn2cncc2C1 S(=O)(=O)(c1ccccn1)N(c1nc(OC)c(Br)cn1)C1CNCC(F)(F)C1 c1(NC(C23C(CN(C(c4ccc(Br)s4)=O)C2)C3)=O)cccc2cccnc12 c1(OC)ccc(Cl)c(C(=O)NCC2CC(F)CN(Cc3ccsc3)C2)c1F N1(C(=O)CN2CCSCC2)CCOC(C(=O)NC2COCC2CO)C1 c1(CC(=O)NC23CC(NC(C(CCC)F)=O)(C2)C3)ccc2ccoc2c1 C#CC1CCN(C(=O)C(CNC(=O)C(C)SCCCC)CC2CCCC2)C1 C(=O)(CCCC(F)(F)CO)N1C(CNC(C23OC(C)C(CC2)CC3)=O)CC1 C(=O)(CC1COc2ccccc21)NC1CC(CNC(Cc2cn(C)nc2)=O)C1 C12(C(N3C4CC(CNC(CC(C)C)=O)C3CC4)=O)CC3CC(CC(C3)C1)C2 N1(C(C(C)c2cccs2)=O)CC2CCC1CC2NC(=O)CCC(N)=O C1(CNC(C2C3CC4C(C3=O)C24)=O)C2CCCC1N(C(c1ccccc1Cl)=O)C2 S(=O)(=O)(c1ccc(Cl)cc1F)NC(C(=O)NC(CNC(C=C(CC)C)=O)C)C C12(NC(C(CC)SC)=O)CN(C(c3cnccc3Cl)=O)CC1CS(=O)(=O)C2 c1(OC)cnc(C(N2CC(F)(CNC(=O)CCn3ncn(C)c3=O)C2)=O)nc1 CC1CN(C(=O)Cc2ccn(C)n2)CC1(C)C(N1CC(C2CCCO2)C1)=O CN(S(=O)(=O)N1CC(O)C1)Cc1cc(F)cc(Br)c1 c1(C(N2C3CC(NC(C4(C(N)=O)CC4)=O)C2CC3)=O)ccc2c(c1)CCOC2 C(=O)(C1CCc2nccn21)NC(C)(CNC(c1cnn[nH]1)=O)C1CCC1 Cc1cccn(CC(N2CC3(CC3)CC2CNC(=O)CN2CC=CC2)=O)c1=O CS(=O)(=O)c1cc(C(=O)NCC2CCC2NC(=O)Cc2ccccc2)ccc1F C1(OC)CN(C(c2cccc(Cl)c2)=O)C(C)(CNC(=O)C(C)(F)F)C1 N1(C(C(CC)SC)=O)CCC2(CC1)CCN(c1cc(CC)ncn1)CC2 C12(CNC(C3CCCO3)=O)CC1CN(C(=O)CCc1nc(-c3ccsc3)no1)C2 C1(C(=O)OCc2ccccc2)CCCN(C(c2cncc(-n3ccnc3)n2)=O)C1 Cc1cccc(Cn2cc(-c3[nH]nnc3C)nn2)n1 CCCCCCN(C(=O)C(O)C1CCC1)CCNC(=O)CN(C)C1CC1 C(C(C(=O)NC(CNC(c1ccc(Cl)nc1N)=O)CC)C(C)(C)C)OCC=C C1(C(N2CC3CCC(C2)C3CNC(C2(CF)CC2)=O)=O)COc2ccccc2C1 C1(C(=O)NCC(CO)NC(CCC)=O)(COC)CCCCCC1 CC(CN(C)N1CCOCC2(CCOCC2)C1)C1CC1 C1(C(=O)NCC(C)(C)OCCN(C)C)(COC)CC=CC1.C12CCC(O1)C(=O)N2 c1(CC(N2CCC(N(C(=O)C(C)N(CC)CC)CCC)C2)=O)ccc(Cl)cn1 C(=O)(C(C)CC(F)(F)F)NC1C(O)CCN(C(CCc2scc(C)c2)=O)C1 N#Cc1ccc(OCC(=O)Nc2cc(N3CCCC3)nc(Cl)c2)nc1 C1(NC(C(c2n(C)ncc2)O)=O)CCCCC1Oc1ccc(O)cc1 C1(C(=O)NCC2C(NC(c3ccnc(C4CC4)c3)=O)CCCC2)CCCC12CC2 N1(C(C(CC)NC(N)=O)=O)CCC2(C1)CN(C(c1cncc(F)n1)=O)CC(C)O2 c1(C(=O)NCC(CNC(C(C)Cn2ccnc2)=O)O)ccc(F)c(Cl)c1F C(=O)(C1=C(Cl)CCC(C)C1)NCCCN(C(CCN1CCC(C)CC1)=O)C c1(C(N2C(C)(c3cn(CCO)nn3)COCC2)=O)cc2ccncc2cc1F N1(C(C=CCC)=O)CC(N(C)C)C(CNC(=O)CC2CCC(C)(C)O2)C1 C1(C(CNC(C(C=C)C)=O)C)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1 C1(NC(c2ccccc2)=O)CCC12CCN(C(=O)CCN1CCCCC1)CC2 c1(C(N2C(CNC(c3cc(C4CC4)no3)=O)COCC2)=O)cc(F)ccc1O c1(C(=O)NC(C2CCN(C(c3cncc(O)c3)=O)C2)C)ncc2cc(Cl)ccn12 C1(C(N2CC(NC(c3ccc(C)c(Cl)c3)=O)C(F)C2)=O)CCC2C(C1)C2(F)F N1(C(c2csc(C)c2C)=O)CC(=O)NCC1C(=O)Nc1cccc(C(N)=O)c1 CCCC(C(O)C(=O)N(C)Cc1cnn[nH]1)NC(c1coc(C)n1)=O C1(NC(c2ccccc2)=O)CC12CCN(C(=O)C(O)CC(F)F)CC2 c1(C(=O)NCC(C)(C)NC(C(C)c2ncco2)=O)cc(Cl)cc2cccnc12 c1(C(C)=O)ccc(C(C)SCC(=O)NCCCNC(=O)Cc2scnc2C)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC(C1CCCCC1)(C)CO C1(C(=O)NC2(CNC(C3C4CC5C(C4)C35)=O)CCCC2)CCCNS1(=O)=O C1(NC(C)=O)CC(NC(=O)NCCS(=O)(=O)N2CCCC2)C1(C)C C(C(O)CC(F)(F)F)NC(CC1N(C(C2CCN(C)CC2)=O)CCCC1)=O N1(C(CCCOC)=O)CC(NC(C2CCCC(F)C2)=O)C2CCCC12 c1(OCCC(=O)NC2CN(C(c3ns[nH]c3=O)=O)C2)ccc(Cl)cc1 C(=O)(C1CCCc2ncnn21)NCC(C)CNC(C1CC(C)(C)CC(C)(C)C1)=O Cc1cc(F)c(NC(C2C3CN(C(c4ccc5scnc5c4)=O)CC23)=O)cc1F c1(C(N2CCC(C)(NC(C3CC4(F)CC3C4)=O)C2)=O)cccc2occc12 CC1CCc2ncc(C(=O)NCC(C)(C3CC3)NC(c3cc(C#N)c[nH]3)=O)n2C1 C(CC(C)C(=O)NC1CC(C)(C(=O)NC2(C)CS(=O)(=O)C2)C1)OC CCC(O)CC(=O)N1CC(O)CC1c1cn(-c2ccc(Br)nc2)nn1 N1(C(CCCC#C)=O)CC(=O)NCC1C(=O)NCC(C)(C)CC(C)C N1(C(C=C)=O)CCCC(CN(C(=O)C(CC)c2ccccc2)CCCC)C1 N1(C(C(c2cccs2)SC)=O)CCC(C2CC2)(NC(c2cc(C)cs2)=O)C1 C(CC(C)(C)C(=O)NCC1CCOC1C(=O)N(CCC(C)C)CC(C)C)SC c1(NCCSc2c(C)cccc2)[nH]c(=NCC2(C)CC(C)(C)C2)nc2scnc12 c1(C(=O)NS(c2cn(C)nc2C(F)(F)F)(=O)=O)ccc2ncccc2c1Cl Cc1cc([N+](=O)[O-])ccc1NCC1CCCC(NC(C2CC(C)C2)=O)C1 CCC(c1ccccc1)=CC(N1CCCC1c1ccc(Br)c(F)c1)=O c1(C(N(CC)CC2(C(C)NC(=O)NC)CC2)=O)ccc(C(=O)O)s1 C1(C(N(C(C)C)Cc2cn[nH]c2)=O)CN(C(c2ccnc(CO)c2)=O)CCC1O c1(CC(N2C(C)(CC)CC(NC(C3CSC3)=O)C2)=O)c[nH]c2c(C)cccc12 C=CC1(C(=O)NCCc2cnn(C)c2)CCN(C(=O)C(O)CC(C)C)C1 C12(C(=O)NCCN(C(C34CCC(C3)C4)=O)C3CC3)CC3CC1C2C3 C1(NC(c2c(CCC)[nH]cc2)=O)CC2(CCN(C(=O)C(n3cc(C)cn3)C)C2)C1 C=C=CCCC(=O)NC(c1nocc1C(=O)N(C1CCOC1)CC)C C12(C(N3CCC(C)(NC(c4c[nH]cc(F)c4=O)=O)CC3)=O)CCCCC1C2(F)F C#CC1(N(C)C)CN(C(C2CCN2C(c2ccc(OC)cc2)=O)=O)C1 C1(COC)CC(O)C(O)CC1C(=O)NOCC(O)CO.c1(C=O)c(C)csc1C C1(C(N2CCCC(CCNC(CC(=C)C)=O)CC2)=O)CC2(CCC2)CCO1 c1(C(N2C(C(=O)NC(CC)CN3CCCCC3)CC2C)=O)cc(C)nc(C)n1 c1(C(=O)NC(C2N(C(c3c(CC)occ3C)=O)CCC2)C)ccc([N+](=O)[O-])o1 c1(OC)ccc2c(n1)N(CC1(c3c(F)cccc3Cl)CC1)CC2 S(=O)(=O)(c1cccnc1NCC1CC(O)CN1C)NCc1n(CC)c(C)nc1 C=CCC(C(=O)NCC1(CNC(=O)C=CC(F)(F)F)CC12CCC2)C(C)C C(=O)(C1CCCc2nncn21)NCC=CCNC(=O)C1=CC(O)CCC1 N1(C(C2(C#C)CCC2)=O)CCC(N(CCO)C(c2nc(C3CC3)cs2)=O)CC1 N1(C(c2cc(C(C)=O)oc2)=O)CC(CN(C(c2cccs2)=O)CC)CC(C)(C)C1 CCCC(C(=O)NC1CN(C(C2CC(=O)N(C)C2)=O)C1)S(N)(=O)=O CCCCC(CC)C(=O)N1CCC(COC)(NC(C2CN3CCN2CC3C)=O)C1 N1(C(c2cn(C)nc2C(F)F)=O)CC(NC(c2ncn(C)n2)=O)CC2(CCC2)C1 c1(OC)ccc(Cl)c(Cl)c1C(N1CC2CCC1C(NC(=O)C(F)=C1CCC1)C2)=O CC(C)C(C(=O)N1CC2CC1(C(=O)NC(C(N)=O)C1CC1)C2)NC(N)=O N1(C(Cn2ncc(C#C)c2)=O)CC(C)(C)CC1C(=O)NC1CC(O)C(O)C1 n1(C(C)C)cc(C(=O)NC(C2CCCCC2)C(C)NC(c2nc(Cl)cs2)=O)cn1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(=CCNC(c2cccc(O)n2)=O)CC1 N1(C(CC2CCC(=O)O2)=O)CCC(CNC(C23CC(F)(C2)C3)=O)C(F)(F)C1 C1(COC(N2CC(C)(C)C2)=O)CCCCN1CCc1cn(-c2cccc(F)c2)nn1 Cc1ccnc(C)c1C(=O)NC1CCOCC1C(=O)NCc1ncsc1C c1(C(C)C)ccc(C(=O)NCCCN(C)C(c2cscc2C2CC2)=O)nc1 C1(C(N(CCCNC(c2cnc(N(C)C)o2)=O)CC)=O)Cc2c[nH]cc2S1(=O)=O Cc1nc(NC(c2nc(C(=O)NCCc3cccnc3)cs2)=O)nc(Cl)c1Br Cc1cc(C(F)(F)F)nn1CC(=O)NC(CNC(=O)C=C1CCC1)C1CC1 c1(OC)ccc(C(C)=O)c(NC(C2CCN2C(C)=O)=O)c1.c1(C(=O)N)ccncc1Br S(=O)(=O)(c1cccc(N2Cc3cnc(Cl)cc3C2)n1)N1C(C)C(O)CCC1 C(=O)(C1=CCC(C)(C)CC1)C(=O)NC12CCCN(C(=O)OC(C)(C)C)C1C2 C#CC1CCC(C(N2CCC(C(C)NC(=O)COc3ccccc3C)C2)=O)CC1 c1(N2C(CNC(=O)Nc3cc(C)nn3CC3CC3)COCC2)cc(Cl)nc(C)n1 C1(C(N(C2CCN(C(=O)C(C)(C)c3ccsc3)C2)C)=O)(CO)CCCCO1 CC1(C)CC(=O)NCC1C(=O)O.C1(NC(=O)Cc2ccco2)CCN2CC12 Cc1ccc(C(=O)C(=O)NCC2CCN2C(=O)Cc2nc[nH]n2)s1 CC(C)(C)CC(C)(C)C(=O)NCC1(C)CN(C(C2(F)CC=CCC2)=O)CCO1 c1(-c2c(F)ccc(OCC)c2F)ccc2c(C(=O)Nc3cnsc3)c[nH]c2c1 C(C(CC(C)C)C(=O)NCC1(CCNC(c2nn(C)c(N)c2C)=O)CC1)OC C1(CNC(C(C2CCN(C(CC3N(C)CC=CC3)=O)C2)F)=O)CC12CCOCC2 C(=O)(CCC1=CCCCC1)N1C(C(=O)NCC(=O)N(C)C)CN(C)CC1 Cc1nc(O)[nH]c1C(=O)NC1CC1CNC(C1(c2ncco2)CCC1)=O C(CCCC(=O)N1CCC=C(C)C1)N(C(C(C)=CCC)=O)C C#Cc1cccc(CC(=O)N(CCNC(c2ccc(COC)c(C)c2)=O)CC)c1 c1(C(N2CCC(C)(C(=O)NCCc3ccsc3)C2)=O)ccc2cc(O)ccc2n1 N1(C(C=C2C(C)(C)CCCC2)=O)CC2CC(NC(c3cncc(F)c3)=O)CC2C1 N1(C(c2c(C)con2)=O)CCC(C(C)(C)C)(CNC(=O)CC2COCCO2)C1 C1(CNC(c2ccc(NC)cn2)=O)CCCCN(C(c2ncccc2Br)=O)C1 CC1=C(C(=O)NC2CN(C(c3snc(Cl)c3Cl)=O)CC2F)SCCO1 c1(NCCSc2scc(N)n2)ncccc1S(=O)(=O)NC1CCOCC1F c1(NC(c2n(CC)nnn2)c2csc(C)c2)ccc(CCF)cc1.C1COCC1 C1(OC)(OC)CCC1C(=O)NC(CNC(c1ccc(SC)o1)=O)CO C1(NC(c2cnn[nH]2)=O)CCC2CCN(C(=O)Cc3csnn3)C12 N1(C(CCCc2onc(C)n2)=O)CC(CNC(=O)C(C)C(F)F)CCC1C C(=O)(C1=C(Cl)CCCC1)NCCC1N(Cc2c(Cl)cn(C)n2)CCC1 C1(NC(c2cccc(CC)c2)=O)CN(C(c2ccc(F)cc2C)=O)CC2CC12 C1(C(=O)NCCC(CNC(C(COCC)C)=O)(C)C)CC2C=CCC(C1)C2 N1(C(C2CC(N(C)C)C2)=O)CCCC2(C1)CN(C(=O)COC1(C)CCC1)C2 Cc1cccc(C(CNC(c2cc(C#N)c[nH]2)=O)NC(c2nscc2C)=O)c1 C1(OC)CC(CNC(C2CCSC(C)C2)=O)N(C(=O)COC2CC=CC2)C1 C(C(C)N=c1ccnc(C2CC2)[nH]1)N(C(C(CC(C)C)C(N)=O)=O)C N1(C(CCn2ncc(C)c2)=O)CCC(CNC(c2nnc(O)cc2C)=O)C(C)C1 CN1C(=O)OC2CN(C(C3(C)C=CCN3C(=O)OC(C)(C)C)=O)CC12 CCCCCCCC(=O)N1CC2CCC2(C(=O)Nc2nccc(Cl)c2I)C1 c1(C(N2CCC(C)(CNC(=O)C(O)C(F)F)C2)=O)c[nH]c2ccccc2c1=O N1(C(CCCOCCC)=O)CC(O)CCC1C(=O)Nc1cccc(OCF)c1 C1(OC)CN(C(=O)C(c2ccc(Br)s2)C)CC1NC(=O)Cc1cncs1 c1(C(=O)NCC=CCNC(c2n3cc(C)sc3nc2)=O)ccc(F)c2c1OCC2 C(C(C(=O)N1CCCCCO1)C(C)(C)C)NC(C1CC(CC)C1)=O N1(C(c2ccn(CC)n2)=O)CC(OC)CC(NC(c2cccc(I)c2O)=O)C1 C#Cc1cc(C(N2CCC(NC(=O)C(C)CCN(C)C)C(F)C2)=O)cc(N)c1 CC1CC(=O)NC1C(=O)NCc1cc(C(N2CC(c3cnccn3)C2)=O)on1 C(C(C)(C)CC(=O)NC(c1cscn1)CO)NC(C(C)(C)CC1CC1)=O C=C(F)C1(CC(N2CC3(CCC3)CC2CNC(=O)CC(C)C2CC2)=O)CCOCC1 Cc1ccnc(NC(C2CCN(C(=O)CC3(O)CCCOC3)C2)C)n1 N1(C(C=C(CC)C)=O)CCC(N(C)C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CC(N2CCCC(C)(NC(=O)CCc3nccs3)C2)=O)CCCC2(CCC2)O1 c1(C(=O)NC(C)C(CO)NC(C2CC(C)(F)C2)=O)cccc(N2CCCCC2)c1 C=C(C)CCCC(=O)NCC1CC(O)(CNC(=O)CCc2cc(F)ccc2F)C1 C1(CNC(Cn2cc(C)c3c2cccc3)=O)CC2CCC(C1)N2C(C1CC1F)=O Cc1cc(=NC(=O)C(=O)N(CC(C)N(C)C(c2ccc3nccn3c2)=O)C)[nH]o1 n1(CC(=O)NC(CC)CNC(c2cnns2)=O)nc2n(c(=O)c1=O)CCOC2 C(C(=O)NCCc1cocn1)(C1CN(C(C2(C)CCC2)=O)C1)OC CCCC(C(O)C(=O)N1CCC(C)(C)C1CO)NC(C1OC2CCC1C2)=O Cc1nc2c([nH]1)CC(C(=O)NCCN(C(=O)CCCCCC(C)O)C(C)C)CC2 c1(C(N(CCCNC(CC2C(OC)CC2)=O)C)=O)nccc2c(C)cccc12 c1(C(=O)NCC2C(NC(CCC=CCC=C)=O)CC2)ccc(C(F)F)cc1F Cc1c(C(=O)NC(C(=O)NCC(C)(F)F)C2CCCO2)ccn1C c1(C(N2CC(C(C)NC(C(C)NC(=O)NC3CCCC3)=O)C2)=O)cnc(Cl)s1 c1(CC(N2CC(OC)C(NC(=O)C(C)CC3CC3)C2)=O)cc2ccccc2s1 N1(C(C2C(C(C)C)C2)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1C N1(C(C2CCC(=O)C2)=O)CCCC(C2CC2NC(c2ccc(F)cc2F)=O)C1 CCS(=O)CC(=O)N1CCC(C(C)NC(=O)C=Cc2ccc(C3CC3C)o2)C1 C#CCC(CC(=O)N(CCNC(c1ccnc(C)c1)=O)C(C)C)c1ccccc1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CC(NC(=O)CC3CCCC3(F)F)C1C2 n1(CC)c(C(=O)NCC2(C)CC(NC(=O)C3=NOC(C)C3)C2)cc2ccccc12 C(=O)(C(C)P(C)(C)=O)N1CC(C)(NC(C(CCC)c2ccccc2)=O)C1 Cc1cc(C(=O)NCCC2CCN(C(=O)CC3(CO)CC3)C2)c(Br)c(C)c1 C(=O)(C(CNC(=O)CCC(=O)N(C)C)C(C)(C)C)N1CCC(C(=O)OCC)C1 c1(NC(C(C2(O)CCC2)NC(=O)COC2CC2)=O)ccc(CCF)cc1 N1(C(C(C)(C)C#N)=O)CC(=O)NCC1C(=O)NC1CC2(C1)CC21CC1 C(C)(CNC(C1CCC1(C)C)=O)(CO)NC(C=CCOC)=O c1(OC)cc(C(=O)C(C)N(CC(C)(C)NC(C)=O)C)ccc1NC(C)=O n1(CCC(=O)NC2CC3(C(NC(c4c(C)noc4)=O)C3)C2)cc(Br)ccc1=O C1(NC(C(C2CCCC2)NC(C)=O)=O)CCCCN(CC(c2nccs2)C)C1 N1(C(c2c(CC)ncs2)=O)CCC2(C1)CN(C(c1cc(C(C)=O)on1)=O)CCO2 Cc1cc(OCC(=O)N(C)CC2CCN(C(=O)C(C)CC(C)C)C2)cc(C)c1 C=CC(C)CC(=O)N1CC(C)(CC(=O)NCCC(C)(O)C2CC2)C1 c1(C(N2CC(C)C(CNC(C3SCCS3)=O)CC2)=O)ccc(F)c(S(N)(=O)=O)c1 C(=O)(C(C1=NOCC1)N(c1ccncc1)CC1CCC1)NCCCC Cc1cccc(CN(C)C(C2(NC(=O)CC3CCCOC3)CC2)=O)c1Cl c1(NC(C2CC(O)CN2S(=O)(=O)CC2CCC2)=O)cc(Br)ncc1[N+](=O)[O-] C(=O)(C(C)CCCC(C)C)N(CCOCCCNC(c1nc(CC)oc1)=O)C S(=O)(=O)(c1cccc(Cl)c1F)N1C(C)(C(N2CCc3c(cccc3F)C2)=O)CC1 c12c[nH]c3c(cc(C(=O)O)cc3c1=O)NC2.Cc1ncccc1CO C1(CC(=O)NC2C(C(=O)NC(c3onc(C)n3)C)CCC=C2)CC(O)C12CCC2 N1(C(c2cc(CC)ncc2)=O)CCCCC(N(C)C(c2cccc(OC)n2)=O)C1 C1(C)(Cc2ccccc2)CCN(Cc2cc[nH]n2)C1.C1C(=O)NN1C n1(C(CNC(COCCCC)=O)C)cc(-c2csc(OC)c2)nn1 N1(C(Cc2c(SCC)cccc2)=O)CCC(CNC(c2ncn(C)n2)=O)C(O)C1 c1(SC)nc(NC2C3CC2CN(C(=O)CC2CCCCO2)C3)cc(Cl)n1 c1(OC)ccc(CC(N2CCC(NC(C3CC(F)(CO)C3)=O)C2C)=O)c(OC)c1 c1(CC)cccc(C)c1C(N1CCC(CN(C(=O)COCCC(C)C)CC)C1)=O c1(CCC(=O)N(CC(C)NC(C2(C)ON=C(C)C2)=O)C)cccc([N+](=O)[O-])c1 N1(c2ncc(C)cn2)CC(NC(C2CCCCS2(=O)=O)=O)CC2(CCOCC2)C1 C1(O)(CN(C)C(C2CC(F)C2)=O)CCN(C(=O)CSc2cn[nH]c2)C1 n1(CC(=O)NCCC(C)N(C)C(C2C(F)(F)C23CC3)=O)nc(Cl)ccc1=O N1(C(C(CC)CC)=O)CCCC2(CCN(C(=O)C(C)n3ccnn3)C2)C1 C1(F)(CNC(c2cncc(C)n2)=O)CCCN(C(=O)C2=CCCCC2)C1 C1(C(N2CC(NC(CCC(C)C)=O)C(F)C2)=O)CCOC2(CCCCC2)C1 C1(NC(c2nn(C)c(O)c2)=O)CC2CCC(C1)N2C(c1cncc(CO)c1)=O C1(CCC(=O)N(C)Cc2ccncn2)CCCCN1C(C1(F)CC(N(C)C)C1)=O C(=O)(C(F)Cc1ccccc1)N1CC(C(=O)NC2CCN2CC(F)(F)F)C1 C(=O)(C1=COCCC1)NC(c1cc(C(C)(C)C)ccn1)C c1(OC)c[nH]nc1C(=O)NCCC1(O)CN(C(=O)CN(C(=O)C(C)C)C)C1 C12(C(=O)NCc3nc(C)c(C)[nH]3)CCCC1N(C(c1nocc1Cl)=O)CC2 N1(C(c2cc(C)sc2C)=O)CCC(CNC(C2CC2c2cccnc2)=O)CC1C N1(C(CCN(CC(C(C)C)C)C)=O)CC(NC(c2nsnc2O)=O)C(N=[N+]=[N-])C1 C=CC(C)N=c1nc2c(ncn2CC)c(NCCCC2CCCCO2)[nH]1 C1(C(N2CC(CC)N(C(=O)Cc3nccn3C)CC2)=O)OCCOC12CCC2 n1(C2(C(=O)NC(C)(C)CCNCC3CC3C3C(OC)C3)CC2)cnc2ccccc12 C1(CNC(c2c(C)[nH]cc2)=O)CC12CCN(C(C13CCCCC1OCC3)=O)CC2 C(CN=C(NCc1cnc(-c2ccccc2)o1)NC1(CC)CC1)OCC=C c1(C(=O)NC2CCC(NC(c3c(C)onc3C3CC3)=O)C2)noc2ncccc12 N1(C(N2C(C(=O)OCC)CC2C)=O)CCC(N2CCC(N(C)C)C2)CC1 Cc1nccnc1C(=O)N(C1CC(NC(c2ccnc(OC3CCOC3)c2)=O)C1)C CC(CC(=O)NCCC1CC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C1)C(F)F N1(C(c2ccc(OC)s2)=O)CCCC(C(=O)Nc2ccnc(Cl)c2)C1 c1(CC(N2CCC3CC2CN3C(c2ccsc2)=O)=O)ccc2nonc2c1 c1(C(NCP(C)(C)=O)C(=O)OCCN2CCOCC2)ccc2c(c1)CCCS2(=O)=O C1(Sc2ccc(NC(N3CC(N4CCCC4)C3)=O)nc2)CCCC(CO)CC1 N1(CC(=O)OCC)CCN(C(=O)CN2CCCC2)CC1.C123CC(C1)(C2)NC3=O c1(C(N2CCC(C(C)NC(CN3CCC(C)C3)=O)C2)=O)cnc2cccnn12 N1(C(c2c(C#N)scc2)=O)CCCC(CNC(=O)CCn2cccn2)CC1 CC(CCCc1ccccc1)C(=O)NC1(c2nc[nH]n2)CCCC1 C1(C(N2C(C)(CCC)CC2)=O)(NC(=O)CC2CC(C)C2)CCCCC1 N1(C(c2c(OC)ccnc2)=O)CCOCC(NC(c2ccc(C(N)=O)nc2)=O)C1 C(CC(C(=O)NC1CC(O)C1O)NC(c1cnc[nH]c1=N)=O)OC N1(C(c2n(CC)nc(Br)c2)C(=O)NC(C)(C)C)CCCC2(CC1)N=N2 N1(C(COC)=O)CCC(CN(c2nccc(CSC)n2)Cc2ccccc2)CC1 CC1COCCN(C(C23COC(C2)C(NC(C2CC2Cl)=O)C3)=O)C1 Cc1ccc(C(F)C(=O)N(CCCN(C(=O)Cc2cnccn2)C)C(C)C)cc1 c1(NC(C2CCCC(NC(c3cc(Cl)cc(I)c3)=O)C2)=O)cc(F)c(Cl)cc1F N1(c2c(C(C)C)cnc(Cl)n2)CC2CCC(NC(C3CCSC3)=O)CC2C1 Cc1[nH]nc(C(=O)NCc2ccc(C(N3CCC(N4CCC4)C3)=O)o2)c1Cl C(=O)(CC(O)CC(C)(C)C)NC(COC)C(=O)NCC(C)(F)C(C)(C)F c1(CC(=O)NC(CN(C(c2cc(CC)n(C)n2)=O)C)C)cccc(CC)c1OC Cc1cnc(C(=O)NC(C)(CO)C(=O)N(CCC(C)(C)O)C)c(F)c1 CCCCC(C)(F)C(=O)NCc1ccc(C(=O)NCC2CC23CC3(F)F)nc1 Cc1cc(Cl)c2c(c1)CCN(Cc1ccc3c(c1)S(=O)(=O)NC=N3)C2 CCC(CO)(C(=O)NC1(CCCC(=O)NC2CC2CCSC)CCC1)OC C1(C(N2CCC(CC(=O)NC(c3nc[nH]n3)C)C2)=O)CC(=O)C1(C)C c1(C(=O)NCCCN(C(=O)CC=Cc2ccccc2)C(C)C)cc2cscc2s1 CC1CN(C(C2C3CCCC23)=O)CC(C)N(C(c2cncc3cccnc23)=O)C1 N1(C(c2cc(C)n(C)c2)=O)CC2CCC1CN2C(c1ccc2snnc2c1)=O C12(NC(c3ccc(CC)cn3)=O)CCCC1CN(C(C1(CCF)CCC1)=O)C2 CCC(C)CC(=O)N1CCC(CC(=O)Nc2ccc(-n3ccnn3)cc2)CC1 Cc1cc2c(cn1)CNC2NC1CC2(C1)CC(C)(C)C2 N1(C(COCC(C)C)=O)CC(NC(c2nc3ccccc3[nH]2)=O)C2(CCC2)C1 C1(C(N2CCCC(NC(c3cccc(CO)c3)=O)C2)=O)CCCC2(CCC2)C1 Cc1cc(C)nc(-c2cn(CC(C)NC(C3(COC)CCOC3)=O)nn2)n1 N1(C(C2(C3N(C(c4cccc(CC)n4)=O)CCC3)CC2)=O)CCC(C)(CC)CC1 N1(C(c2cc[nH]c2)=O)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C2CCC12 c1(CCC)ccc(C(N2CC3CC2C3NC(C2(C3CC3)CC2)=O)=O)cc1N C=C(Cl)CC(C(=O)N(CCN=[N+]=[N-])C)NC(=O)C(C)C1CC1 C1(CNC(c2c(C)ncnc2O)=O)C2CCCC1N(C(C1CC(CCO)C1)=O)C2 C(=O)(CC(CC)C(C)C)NC1CCCC(C(N(CCC)C(C)C)=O)C1 C1(n2c(CC(C(=C)C)OC)nc(-c3cnn(C)c3)n2)CCC(F)(F)CC1 C1(C)(C(=O)OC)CCCN(N2CCC(CN3CCOCC3)C2)C1 C1(F)(C(=O)NC2CC(C)(NC(=O)CCN3CCOC3=O)C2)C2CCCCC12 c1(OC)cc(N)c(C(N2CCC(CNC(=O)CC(C)C)(OC)C2)=O)cc1F c1(N(C2CCN(C(=O)CCCF)C2)C(C)=O)ccccc1.C1(C)C(=O)N1 c1(C(NNC(C2C=CC(=O)N=N2)=O)=O)ccc(OCc2ccccc2)c(OC)c1 C1(C2CC2)(CNC(c2cc(OC)no2)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C1 c1(C(=O)NC(C)CNC(=O)C(c2cccn2C)=O)cc(C(F)F)cc(F)c1 Cc1cc(Cl)cc(Cl)c1OCC(=O)NC(C)CNC(=O)Cc1ccco1 N1(C(=O)NCC(C)S(C)=O)CC2(CCC2)CC1C CC1(C)CCCC(O)(C(=O)NC2CCC2NC(c2cccc3nccn23)=O)CC1 c1(C(N(CC(=O)NCc2cc(OC)ns2)C2CCC2)=O)ccnc(CO)c1 c1(C(N2CCC(CNC(C3(OC)CCC3)=O)C23CC3)=O)cc2ccsc2n1C c1(C(=O)NC2CC(CCNC(C(C)(C)SC)=O)C2)n[nH]c(C)c1Br C1(NC(c2c(C)csc2Cl)=O)CCN(C(=O)CCc2ccoc2)CC1F C(C(=O)OC(C)(C)C)(C(=O)NCC(C(C)(C)C)NC(c1cnncc1C)=O)OC c1(OC)ccc2c(c1)CC(C(=O)NC(C1CCCCC1)C(C)NC(=O)C=CBr)O2 c1(C(=O)NCCC(=C)CNC(=O)CCOC)coc2ccc(C(C)(C)C)cc12 c1(C(=O)NCCCC(N2CCC(CNC(c3c(N)non3)=O)C2)=O)ccc(F)cc1 Cc1noc(C)c1CC(C)NC(=O)CCN(CCCO)C.C12CN(C1)OC2=O N1(C(c2ncc(C)s2)=O)CC2C3CCC(C2C1)N(CC1CCOC(C)C1)C3 Cc1ccc(C(=O)NCCNC(=O)CC(=O)OC(C)(C)C)c2cccnc12 c1(C(N2CC(F)(CNC(C3CCC(OC)C3)=O)C2)=O)cn(C2CC2)nc1C Nc1ccc(C(=O)NCC=CCNC(c2cc(Cl)ccc2F)=O)c2c1CCCC2 N1(C(c2cc(CCOC)no2)C(=O)NCCC2CC2)CCC(C2CCN(C)C2)C1 C1(CCN(C(=O)CC2OCCC2C)C)CCN(C(=O)C2=CCCO2)CC1 C12(CNC(c3n(C(C)C)ccc3)=O)CC(NC(C34CC(C)C3C4)=O)(CO1)C2 Cc1cc(=O)ccn1CC(=O)N(C)CC1(O)CCN(C(=O)Cn2ccnn2)C1 c1(N2CCC(NC(CNS(CC)(=O)=O)=O)C(C)C2)ncnc2c1nnn2C1CC1 C1(CC)CCCN(C(=O)C(C)C2CCCC2)C1C(=O)NC1CC(C(N)=O)C1 N1(C(C=CC(C)NC(c2ccc(SC)o2)=O)=O)CCN2C(=O)OCC2C1 C(C(C)(C)CC(=O)NCc1cc(C(C)C)n[nH]1)NC(C1C(C)OCCO1)=O C1(NC(c2ccc(C)cc2)=O)CN(c2nc(C(F)(F)F)ns2)Cc2nccn2C1 NC(=O)C(F)CC(N)C(=O)N1CCC12C(=O)Nc1ccccc12 N1(C(c2cc(C)n(CC(F)(F)F)n2)=O)CC(C)(C)CC1CO c1(C(N(C)CC2CCCN2S(C)(=O)=O)=O)ccc(CNC(C2(C)CSC2)=O)nc1 N1(C(CCCCCC)=O)CC(NC(=O)C(O)C(C)C)C(C2CC2)C1 c1(CCCC2(O)C3(CNC(C4(OC)CC4)=O)CCC2C3)c[nH]c2ccc(Br)cc12 N1(C(CCC(C)C)=O)CCN(C(C2CN3CCCC3CO2)=O)CC(O)C1 Cc1ccnc(Oc2ccc(NC(c3cc(N(C)C)cn3C)=O)cn2)c1 c1(C(C)(C)C)ccc(CCC(C2(O)CN(C(C3(O)CC3(C)C)=O)C2)(C)C)o1.N c1(C(c2cn(C3CCN(C(=O)Cc4cocn4)C3)nn2)(C)C)cccc(Cl)c1 C[S+](C)CCC(O)C(=O)OC(C12CC(CNC3(C)CCCCO3)(C1)C2)=O C1(C(N2CC(C)(NC(c3c(C(=O)OC)cccn3)=O)C2)=O)CCC2C1C2(F)F n1(CC(=O)N(CC(C)O)CCNC(c2cnoc2)=O)cc(SC2CC2)cn1 C=CC1OCCC1NC(c1nonc1N)=O CC(C)CC(O)C(=O)NCCCCC1CN(C(=O)C(C(C)C)c2cccnc2)C1 C(C)(C)(CC(F)C(=O)N1CCCC1CN=[N+]=[N-])NC(c1c(OC)nsc1)=O CCCC(C#N)C(=O)N1CC(CNC(c2cnc(C3CC3)nc2)=O)C(O)C1 CCC(CC)C(C)C(=O)NC1COCCC1NC(=O)CCN(C)CC CC1(C)CCCOC1CC(N1CC=CC(NC(=O)Cc2ccoc2)C1)=O CC1(C#N)CCCN(C(=O)C(C)(C2CCC2)NC(c2nsnc2O)=O)C1 c1(C(=O)NCC(C(=O)OCC)CC)cc2cc(C)cc(C)c2[nH]1 CC1CC=C(C(=O)N2CC3CC3C2C(=O)NCc2ccnc(O)c2)CC1 C1(C2CCC2)(CNC(CN2C(C)CC2)=O)CCN(C(c2cn[nH]c2)=O)CC1 N1(C(C2C(C)C2C)=O)CCCC(CN(C(=O)Cc2cc(Cl)n(C)n2)C)C1 CC(C)C(CNC(c1csc(O)n1)=O)NC(=O)C=CCn1cncn1 N1(C(c2ccc(C(F)(F)Cl)cn2)=O)CC2CC1CN2Cc1ccccc1 c1(CNC2C(C(N(C(C)C)CCO)=O)C2)cc2ccccc2nc1O N1(C(CC(C)N(C(CSCC)=O)C)=O)CC(C)C(C)C1C Cc1cc2c(C(=O)N(C(C)CNC(C3CCC4(CCC4)C3)=O)C)cccc2o1 c1(C(=O)NCCC(C)NC(=O)C(C)Cc2ccco2)ccc(F)c2cnccc12 c1(C(=O)NCC2CN(C(c3c(C)onc3)=O)C2)cccnc1CC(C)C c1(C(=O)O)cccc(S(=O)(=O)N2CCCC3(CCO3)C2)c1 C1(F)(CNC(c2cccc(F)c2F)=O)CCCN(C(=O)CCC2CCCOC2)C1 C(=O)(CC(C(C)(C)C)NC(C1CC2(CC2)C1)=O)N1CCC(C(C)C)C1 C12(NC(c3ccc(O)nn3)=O)CCC(C1)N(C(=O)Cc1nc(C3CC3)cs1)C2 c1(CC(N)=S)ccc(CNC23CC4CC2C3C4)cc1 C1(NC(C2CCC(C(N)=O)C2)=O)CCC(NC(=O)CC2CCSCC2)CC1 c1(C(=O)NC2CCC(CNC(=O)CC3CCCCC3)C2)cn2cccc(Cl)c2n1 C1(NC(C2CCSC2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2(CC2)C1 C1(C)(C(=O)NC(CCC)CCCNC(c2ccc(C)o2)=O)CCS(=O)(=O)CC1 C1(NC(C2(C(C)C)CC2)=O)CC2(C1)CN(C(=O)CSc1ccccc1F)C2 c1(C(N2C3CN(C(=O)CC4CCCO4)CC2CC3)=O)ccc2c(c1)OC(F)(F)O2 CCC(CCNC(=O)CCCn1cc(CCCOC)nn1)C1CC1 C1(C(=O)NC2C(NC(Cn3nnc(C)n3)=O)C2)CCc2ccccc2O1 N1CC(OC)CC(C)C1.c1(OCC(=O)Nc2c(OC)n(C)nc2)cc(C)ccc1F c1(C(=O)NC2(C)CCN(C(C=CS(C)=O)=O)C2)cc(F)c(Br)cc1F c1(C(=O)NC2CCC(N(C(CCC=C)=O)C)C2)c(C)ccnc1C C(=O)(C1CCCc2n[nH]cc21)NCC1C(C)CCN1C(=O)CCc1cnoc1 c1(C(=O)NCC2(CNC(=O)C=CC3CCOCC3)CC2)cc2cc(O)ccc2[nH]1 c1(C(=O)NC(CNC(C2CCC(=O)N2C2CC2)=O)C2CC2)cc2cnccc2o1 CC1(C#CC(=O)N2CCOC3(C2)CN(C(=O)C#CC2(C)CC2)C3)CCCO1 CC1CC2CCC(C(=O)NC(C)CCCCNC(c3cc(=O)cc[nH]3)=O)CN2C1 c1(C(=O)NC(C2CCCN2C(=O)CCCC2CCCC2)C)ccc(O)nc1 c1(CNC(C2CC(c3ccc(Br)cc3)(O)C2)=O)c(Br)ccc(F)c1F c1(CSC)ncnc2[nH]cnc12.C(CCN=C1NCCN1)C1(OCC)CCCO1 N1(C(c2c(C)onc2)=O)C2CCC1C(CNC(=O)C(C)(O)C1CCC1)C2 Nc1cc(C(=O)NC(CNC(c2csc(Br)c2)=O)CO)cc([N+](=O)[O-])c1 CCCCCCC(C)C(=O)NC1COCC1C(=O)NCCC1(SC)CCC1 c1(CC(=O)NCC2C(NC(C(C(C)C)SC)=O)C2)cn2cccc(C)c2n1 c1(-c2n(-c3c(C(C)C)cccc3)nc(-c3ccc(N)cc3)n2)ncc(F)cc1N c1(OCC)ccccc1CCC(N1CCCC1(C)C(=O)Nc1cccnc1O)=O CC1CCC(CNC(=O)CN(S(C)(=O)=O)C)N(C(=O)Cc2cccc(F)c2F)C1 C1(CCCC)CN(C(C2NC(=O)C3CC23)=O)CCN1C(=O)C1=CCCC1 CCCC(CC)CC(=O)N1CCC(Cn2cc(-c3nccs3)nn2)CC1 c1(CC)ccccc1C(=O)NC1(C)CCN(C(=O)CC2CCOC(C(C)C)C2)C1 c1(CC)cc(C(=O)NCC23CC(NC(C4CCCN4C(C)C)=O)(C2)C3)c(C)nn1 c1(C(c2n(CCOCC)nnn2)NC(c2ccn(C)n2)C)ncc(F)cc1F C1(NC(CSCCNC(CCc2cc(C)[nH]n2)=O)=O)CC(O)CC1O Cc1cnccc1C(C)C(=O)NC1CCCCC1N(C)C(c1cccs1)=O C1(C(N2CCN(c3ncc(C)c(C)n3)C(C)C2)=O)CCOC2(CCCC2)C1 c1(CC)cc(NC(=O)Nc2ccc(Br)cc2OC(F)F)ccc1OC(F)F n1(CCC(=O)NCC(CC=C)NC(c2c[nH]nc2C(C)C)=O)cnc(C)cc1=O C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(NC(=O)CC(C)(C)CN(C)C)CC(C)C1 C=C(Br)CC(=O)NC(C)CCNC(c1n[nH]cc1C1CC1)=O C12(C(=O)NC(C(=O)OCC)CCc3ccccc3)CCC(CC)(C1)OC2 Cc1cc(C#N)nc(NC23CCCN(C(c4occc4C4CC4)=O)CC2C3)n1 c1(C(=O)NCCc2nnc(C)o2)ccc(S(=O)(=O)N2CC(C)(N(C)C)C2)o1 c1(C(C)OCC)cn(CCOCCNC(=O)CCn2ccnn2)nn1 c1(C(=O)O)cncc(-n2cc(C3CCCN3C(=O)C(C)c3cncs3)nn2)c1 c1(C(=O)OC)ccc(N2CC(CCCCNC(c3cnc[nH]3)=O)C2)nc1 c1(OC)ccc2c(c1)C(CCNC(c1cccc(C)c1)C1CCCCC1)=CC2 N1(C(CN(c2ccccn2)C)=O)CCC(O)(CCNC(=O)C(C)(C)N(C)C)C1 CCCN=C(NCC1(CO)CC1C(F)(F)F)N1CCC(F)(c2ccncc2)CC1 c1(NC(c2n(C(CC)C)nnn2)c2ccc(C(F)F)o2)ccc2nncn2c1 C#CCC(O)C(=O)NC1CC(NC(=O)C(F)(F)c2ccsc2Cl)C1 N1(C(C(CNC(c2c(OC)ccnc2)=O)C)=O)CCOCCC1C(C)C C(=O)(C#CC1CCC1)NC1C(CNC(c2c(COC)cccc2)=O)CCCC1 C1(C(N2CCC3(NC(C=C(CCC)C)=O)C(C2)C3)=O)CC2(CC(C)=NO2)C1 N1(C(c2cnnc(Cl)c2)=O)CC2CCC1CN(c1ncc3ccccc3n1)C2 O=C(C(C1=NOCC1)N1CCCC1c1cccc(Cl)c1)NCc1ccc(F)cc1 N1(CC(=O)NC(CN(C(=O)CNC=O)C(C)C)C)C(=O)c2ccccc2S1(=O)=O c1(OC)c(C(N2CC=CC(NC(=O)CC(C)N(C)C)C2)=O)[nH]c2ccccc12 [N-]=[N+]=NC1CN(C(c2cn3ccnc3s2)=O)CC1NC(c1ccc([N+](=O)[O-])[nH]1)=O c1(C(N(CC(=O)Nc2ccc(OCC(=O)OC)cc2)C)=O)cc2ccsc2cn1 c1(CCNC(Cc2c(I)ccc(C)c2)=O)cc(Br)c2c(c1)CCO2 c1(OC)ccc(CN2CCNCC2C(=O)NCc2ccc(Br)cc2)c(Br)n1 N1(C(CC=CCC)=O)CC2CCC(C1)N2C(=O)Cc1nnc(S)n1C c1(CC)c(C(N2CC(CC(C)NC(=O)CSC(F)F)C2)=O)oc2ccccc12 N1(C(C2(C(=O)OCC)CC2)=O)CCCN(C(=O)CC2CC(C)N(C(N)=O)C2)CC1 N(C(=NCCCF)NC1CCN(c2nnc(C)n2C)CC1)C(CC)CC C12(NC(CNC(COC)=O)=O)CCC(C1)N(C(=O)CCOC1CCCCCC1)C2 C1(C(N(CCOC)CC2CC2)=O)C2CC(O)C(C2)N1C(C1CC(C)CO1)=O c1(OCCCC(=O)NCCN(C(C2C(CCOC)C2)=O)CC)cccc(C)c1C c1(NC(c2ccnc(C)n2)=O)ccc(NC(c2scnc2C)=O)c(F)c1 c1(C(=O)NC2C(CC)C2)cc(NC(c2cc(C(F)F)[nH]n2)=O)ccn1 C(CC(C(C)(C)C)NC(=O)C1=C(Cl)CC1)N(C(CCCN(C(C)C)C)=O)C C1(CNC(C(C)NC(CC)=O)=O)CN(C(=O)C(O)C(C)C)CCC1C(F)(F)F C1(CC(F)F)(C(=O)NCCCC(C)NC(C2CCC(C)(C)O2)=O)CCOCC1 C1(C)(CNC(c2cc(C(C)C)nn2C)=O)CCN(C(C2CC2(F)Cl)=O)CC1 N1(C(C=CC=CC)=O)CCCCC1C1CCN(C(=O)C(C)n2cnnn2)CC1 N1(C(C(C)OC)=O)CCN(C(=O)C=CSc2nc[nH]n2)CC(C)(F)C1 C#CC1(CNC(=O)C(CC(C)C)NC(=O)CCCSCCC)CCOCC1 c1(C(=O)NCC2(CO)C(C)(C)C2)cc2occc2[nH]1 C1(CN(C(CC2CC(CC)C2)=O)CC)CN(C(=O)C(C)(C)CC2CC2)CCO1 C1(CNC(=O)COC(F)(F)C(F)(F)F)CCCCC1NC(=O)CN1CCOCC1 Cc1cc(C(N2CC3(NC(c4cc(C(C)C)[nH]n4)=O)CCC2C3)=O)cc(C)c1N C1(CNC(c2c(C(C)C)ccs2)=O)CCC2(CN(C(c3[nH]ncc3C#N)=O)C2)O1 C1(NC(C=CC(=O)N(C)C)=O)(CF)CCN(C(C2COC(=O)O2)=O)C1 CN1CC(O)CCC1C(=O)N(CC(N1CC2CC2C1)=O)C1CC1.n12cc(nn1)C2 N1(C(c2ccoc2CNc2ccc(Br)nc2F)=O)CCCCCC1C=O.CCO N1(C(CCc2ccc(C)o2)=O)CCC(F)C(NC(c2nc(C)oc2C)=O)C1 c1(C(C(=O)NCC(C2CC2)NC(C2(C)CC2(F)F)=O)(C)O)ccccc1F c1(C(=O)NC(CN(C(=O)CC(C)SC)CC)C)nnn(C)c1N Cc1ccc(C(=O)NCCCC2CCCN2C(C23COCC2C3(F)F)=O)nc1C C(=O)(CCCN(C(=O)CC1(N(C)C)CC1)C)N(C)Cc1cscn1 C(=O)(C1COc2ccccc21)N(CC(C)N(C(c1cc(OC)c(O)nc1)=O)C)C C(CCCC(C)NC(c1c(C)coc1C(C)C)=O)NC(c1cnc(CC)[nH]1)=O CCC(S(=O)(=O)N1CCN(c2ccccn2)CC1)c1ccccc1 C1(C(=O)NC(COC)C)CN(C(C2CCCCC2C(C)(C)C)=O)CC1(F)F C(=O)(C1=C(C)CCCC1)N(C1CCN(C(c2cc(C(C)=O)[nH]n2)=O)C1)CC C1(OC)C(NC(C2CC(C)N2C(c2ccoc2C)=O)=O)CC1O N1(C(c2n(CC)ccn2)=O)C2CCCC1CC(N=c1[nH]c(Cl)ncc1C(C)C)C2 N1(C(C=Cc2cn(C)nc2)=O)CC2CCCN(C(C34COC(CCO3)C4)=O)C2C1 N1(C(c2nc(C(C)OC)oc2)=O)CCOC2(CCCNC2)C1 c1(NC(C)=O)ccc(O)c(C(=O)NCC2OCCN(C(CSCC(=O)OC)=O)C2)c1 c1(CC(N2CCC(O)(CNC(c3cnn(CC)c3C)=O)C2)=O)cc(C)cc(F)c1 c1(C(N2CCC(CN(C(=O)C(C)(C)C)C)C2)=O)cccc2c(O)nncc12 c1(C2(CNC(c3cc(OC)ncc3)C)CC2)cccc(OC)c1OC N1(C(c2cccc(NC(C)=O)c2C)=O)CC2CCCC2(Nc2cnc(C#N)cn2)C1 CC(CC(=O)NC1(CNC(c2ccccc2C2CC2)=O)CC1)C(F)F C1(COC)CCN(C(C2CCCCC2NC(=O)CCc2ccccn2)=O)CC1 C(C)(CC(C)NC(=O)Cc1csc(-c2ccncc2)n1)NC(C(C)SC)=O N1(c2nc(COC)nc(C)c2)CC2CCC1C1CN(C(C3CC3(C)Br)=O)CC21 C1(C)(CNC(C2CCN(C)C2)=O)CCCN(C(=O)CCCNC(=O)C(C)(C)C)C1 N1(C(Cc2c(C)ccnc2)=O)CCC(C)(C)C1CC(=O)NC1CC2CCC1O2 C1(NC(C=CC(CC)C)=O)CCN(C(=O)Cn2nc(C(F)(F)F)cc2C)CC1O CC(C)(CC#N)C(=O)NCC(C1CCOC1)NC(C1(C2CC2)CCC1)=O C12(NC(C(CCSC)O)=O)CCCC(NC(=O)CCc3ccc(N)cn3)(C1)C2 c1(C(N2C(C)CC(CNC(COCC)=O)C2)=O)cc(Br)cc2c1OCO2 C(=O)(C1=CCCCC1C)N(CCCNC(=O)C(c1ccc(OC)cc1)OC)CC C(Cc1ccc(Cl)cc1)(C(F)(F)F)(c1ccccc1)N(CC(C)C)C N1(C(COCC=C)=O)CCC(C)C(CNC(=O)Cn2cccn2)C1 CC(C)CC(c1ccccc1)NC(=O)NC(C1CCCO1)C(C)C1CC1 C(=O)(C(Cc1cn[nH]c1)NC(C1CCCCC1)=O)N1CC(C(C)OC)C1 CC1(C)C(=O)CC1C(=O)NOCCCCC1CC1.C1(CCNC=O)(CO)CCCC1 C(=O)(C#CC1CCOC1)N1C(CNC(c2ccnn2CC2CC2)=O)CCCC1 c1(OC)ccc(=NC(C)c2cn3ccccc3n2)[nH]n1 N1(C(C)=O)CCCCC1C1CCCN1C(=O)CCNC(c1cn(C)nn1)=O c1(C(N2CC(CNC(CSCCCC)=O)C3C2C3)=O)cnc2[nH]c(=N)sc2c1 C=C(C)CC(C(=O)N=c1ccn(C(F)F)[nH]1)NC(=O)C(C)CSC CCS(=O)(=O)c1cccc(C(=O)NC(C)CNC(=O)C=C2CCSCC2)c1 N1(C(Cc2nc(NC=O)sc2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C2CC12 c1(C(=O)NCC2CCCCN2C(=O)CN2CC=CC2)csc2ccncc12 c1(OC2CN(C(CSC)=O)C2)ccc2ncccc2c1.C12(CCCC1)C(=O)NC2 Cc1cc(=NC(=O)C(C)NC(c2cc[nH]n2)=O)[nH]n1C C(C(C)CC(=O)N1CCCCC1C(=O)NCCS(C)(=O)=O)OC N1(C(CC(CC)CN(C)C)=O)CCC(NC(c2cc(CO)[nH]n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(F)cc1)NC(c1ccccc1)CNC(N1CCCC(C)C1)=O C1(NC(C2C(OCC)C2)=O)CCCN(C(c2cc[nH]c2C)=O)CC1 CC(C)(CC(=O)NC(CC1CC1)CO)NC(C1CC1C(F)F)=O CCC1=C(C(=O)N(CC(C)(C)O)C2CC2)CCCO1.C1(C)C(=O)N1CC N1(C(CCCC(=O)NCC)=O)C2CCC1CN(C(=O)C(C)C(O)CC)C2 C1(C(=O)NCc2cc(C)no2)C(C)OCCN1C(=O)C(C)CC(N)=O N1(CC)OCC(NC(=O)CC2(C)CCN(C(C3CCC3C)=O)C2)C1=O CC1COCC(C(=O)NC(C(=O)NCCC2CC=CC2)C(C)O)O1 c1(C(=O)NC2CN(C(=O)CC3OCCO3)CC2O)n[nH]c2ccc([N+](=O)[O-])cc12 c1(C(=O)NC2CC(OCC(=O)NCC3CSCCS3)C2)cccc(O)c1 c1(C(N(C2CN(C(C(C)OCC#C)=O)CC2(C)C)C)=O)cccc2nn(C)nc12 N1(CC(CC(C)C)N(C)C)CCC23CCC(CC12)C3(C)C c1(C(=O)NC(c2cncc(C)c2)CO)ccc2cnc(C)n2c1 c1(CC)onc(C(=O)NCCCCCn2cc(C3(O)CCCC3)nn2)c1C C1(NC(CCCCCC)=O)CN(C(C2CSCCS2)=O)Cc2ccnn2C1 C(=O)(C(C)(C)CC(=O)NC(C)(C)CNC(=O)CCN1CCC(F)C1)OC N1(C(CN(C(=O)OC)C)=O)CCC(NC(=O)C(C)CC(F)(F)F)C12CCC2 C=CC(C)CC(=O)N(C)CC1CN(C(c2coc(C(C)(C)C)n2)=O)CCO1 S(=O)(=O)(c1cnc(Cl)nc1)N1C(C(N2CC3CC3C2)=O)CC2CC21 C1(CNC(c2ccc(F)c(CO)c2)=O)CCCN(C(C2CC2C(F)F)=O)CC1 c1(C(N2CCC(NC(c3ccc(CSCCC)o3)=O)C2)=O)cncc2c1CCC2 c1(C(=O)NCc2c(C(=O)NC(C(=O)OCC)C3CC3)cco2)cc(C)c(O)nn1 C1(O)(CCNC(C=Cc2ccc(C)s2)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 c1(OC(N(c2ccc(N3CCCC3)nc2)C(CCC)=O)=O)ccc2cc[nH]c2c1 C1(CNC(N2C(C#C)CCCCC2)=O)CCCCC1C1CC1 Cc1ccc2c(c1)CCC(C(=O)N(c1ccccc1)Cc1ocnc1C(=O)O)O2 N1(C(C(=O)NC2(C)CC2)c2ccns2)CCOCCC1C(C)(C)C N1(C(C23CC(OC)C2C3)=O)CCC(NC(=O)C(c2cccn2C)=O)CC1 CCC(C)CC(=O)NCC1(c2ccccc2)CC(NC(=O)CCN2CCC2)C1 C(=O)(N=c1[nH]n(C)c2ccc(Cl)cc12)c1cncc(NC(CCCC(C)C)=O)c1 c1(C(=O)NCCCC(C)NC(C2(Cl)CC2)=O)cccc(C2CCC2)n1 c1(OC)cc(CC(N2CCC(O)C(NC(c3cocc3C)=O)C2)=O)ccc1C Nc1cc(Br)ccc1C(=O)NCC1CN(C(=O)C(O)C(F)F)C1 C1(NC(CC(C)F)=O)CN(C(c2ccc(Br)cc2)=O)CCC12CCC2 N1(C(CC(=C)Br)=O)CC(CNC(c2ccc(OC)nn2)=O)CC12CCC2 C(CN=c1nc(N(C)CCF)c2c([nH]1)CSC2)c1ccc(C)c(F)c1 C1(CNC(c2ccc(C3(O)COC3)cc2)=O)CCN(c2ccnc(CO)n2)CC1 C1(C2C(NC(C=CC(=O)N(C)C)=O)CCO2)CCN(C(=O)CC2CCSC2)CC1 C(=O)(C1Cc2ccc(F)cc21)NCC1(NC(C(COC)OC)=O)CCCCC1 c1(OC)cc(CC(=O)NC(C(C)NC(C23CC(F)(C2)C3)=O)C(C)C)ccc1Cl N1(CCCC)CCCCC1C(N1CCC(F)(CNC(c2coc(C)n2)=O)C1)=O C(=O)(CCC(=O)NC)N(C1CCCN(C(=O)C=CCN2CCCC2)C1)CC c1(C(C(=O)NCCS(CC)(=O)=O)NC(=O)Cc2cc[nH]n2)c(C)cccc1Br C12(C(N3CC(c4cc(O)no4)C3)=O)COCC1CN(CC1CC3CCC1CC3)C2 C(=O)(C(C(C)CC)SC)N(C12CC(C1)C2)CC C(C1=CCN(C)CC1)(c1nnnn1-c1ccc(F)cc1)NCc1ccc(OC)nc1 C1(CCNC(C(CC)Oc2ccccc2)=O)CCN(C(=O)C(C)(C)COC)CC1 Cc1cc(Cl)ccc1CN(c1cc(CN)ccc1C)C.C12CN(C1)C2=O c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nccn2)cc(F)ccc1Cl C(=O)(C(F)C(C)(C)O)N(CCC(=O)NCCCN1CCOCC1)C(C)C C1(C(C)(C)C)(CNC(c2ccc(C(C)=O)s2)=O)CCN(C(c2cnnn2C)=O)C1 c1(NC(C2CCC(CCC)N2C(=O)C(C)n2ccnn2)=O)cc(F)c(O)cc1C n1(CC(=O)NC2C(CNC(CC3(C)CCCCC3)=O)C2)ccc(O)nc1=O Fc1ccc2c(c1)C(c1nc(-c3cccc(Cl)n3)nn1C1CCCSC1)C2 n1(C2(C(N(CCCNC(C3CC(O)C3)=O)CCO)=O)CC2)cc(Br)cn1 c1(NC(CC)CNC(=O)Cc2ccsn2)nccc(-c2ccccc2)n1 C(=O)(C(C(C)(C)C)NC(N)=O)NCC(C)NC(C(C)CC1CCCC1)=O C(=O)(C1CCCc2cncn21)N1CCCC2(CN(C(C3C(=C)C3)=O)C2)C1 N1(C(C2(C=C)CCN(C(C3OCCCC3(C)C)=O)C2)=O)CC(OC)C(C2CC2)C1 c1(C(=O)NC(CNC(C2C(C)C2C)=O)C(C)(C)C)ncc2ccccn12 O=C1CCN(CC2OCCO2)C(=O)N1CC1(c2ccsc2)CC1 c1(OC)ccc(NC(=O)C(C2CCN(C(C3CCCO3)C)CC2)C)c(C)c1 c1(C(=O)NC2C(NC(c3cc(C)c(O)cc3)=O)CC2)cc(P(C)(C)=O)cs1 C1(C(C(=O)NC2(CC(N)=O)CCC2)NC(c2cn[nH]c2)=O)CCCCC1 c12ccccc1OC2=O.n1(CCOC)cnnc1C(=O)NOC(CC)CC c1(OC)ccccc1OCC(=O)NC1C=CCN(C(C2C=C2C)=O)C1 O=C(CCCCCF)NCC1C2CC1N(C(=O)Cn1ccc(C3CC3)n1)C2 N1(C(C2CSCCN2C(C2CC2C(F)F)=O)=O)CCCC2(CC(O)C2)C1 c1(N2CCCC(CC=CC)C2)nc(N2CCC(C)(C3CC3)C2)c2ccsc2n1 Cc1cccc2c(CN3CCC(NC(=O)CCCCCBr)C(O)C3)c[nH]c12 c1(C(=O)NCCN(C(c2ccc(F)cn2)=O)CC)cccc(C)c1O c1(CN(C(=O)CNC(=O)CC2CC2)CC)cccnc1 C1(CC)CCN(C(=O)COC(C)(C)CC)C1CNC(=O)CCC1CC1 Cc1c[nH]c2ncc(C(N3CC(NC(c4cc(C#N)c[nH]4)=O)C(C)(C)C3)=O)cc12 C1(NC(c2cnc(OC)c(Cl)c2)=O)CCN(C(c2sccc2Cl)=O)CC(C)(C)C1 Cc1ccc(C(=O)Nc2nc(-c3ccc(C(F)(F)F)nc3)cs2)c2cccnc12 C#CCCCC(=O)NC(c1ccccc1Br)CNC(=O)CSCCC C1(CO)CCC(N=c2nc(N3CCC4(CCCCCC4)CC3)c3sccc3[nH]2)C1 C1(NC(COC(C)=O)=O)CCC(N(C)C(c2sc(Cl)cc2Cl)=O)CC1 c1(NC(C2(C(C)(C)C)CCNC2)=O)cc(C(=O)O)c(Cl)c(F)c1 Cc1cccc2c(C(=O)NCC3CC4CCC3CC4)c[nH]c12 Cc1ccc(Cl)c(C(=O)NCC2(O)CCN(C(=O)C(C)C3CCCC3)C2)c1 c12cc([N+](=O)[O-])ccc1N1CC3(CN(C3)C2=O)C1.C(C(O)C(=O)OC)OC C1(NC(C=C(C)C(C)C)=O)CC(c2ccccc2)CO1 N1(C(C=CC)=O)CCC(NC(=O)CSc2nnnn2C)CC1c1ccccc1 N1(C(C2CC23CCCC3)=O)CCCC2(CCCO2)C1 C1(N)C2CCC(C2)C1CO.C1(N)CC(NC(CNC(COC(C)=O)=O)=O)C1 C1(CC#C)(C(N2CC(OCCNC(=O)CCc3cccnc3)C2)=O)CCCCO1 c1(N2CCN(C(C(=O)NCCCC)COC(C)(C)C)CC2)nsc2ccccc12 C(=O)(C#CC1CCOC1)N(C(C)C(=O)NC(C)(C)CN1CC2CC2C1)C1CC1 c1(CCCC(=O)N(CC(C)(C)NC(C(C)C(C)(C)C)=O)C)nc2ccccc2[nH]1 C1(O)(CCNC(=O)Cn2cnnc2O)CCN(C(=O)COC2CCOCC2)C1 CCCC(CC(=O)NC(C)C(N)=O)NC(C1C=CCC1)=O N1(C(c2cc(C)[nH]n2)=O)CCC(C)(C)C1CC(=O)N(C1CCCC1O)C1CC1 Cc1cc(Br)ccc1C(=O)Nc1c[nH]nc1C(=O)NC12CC(C(F)(F)F)(C1)C2 CC1=CC(C)CN(C(=O)NCc2cccnc2N(C)C)C1 c1(C(N2CCN(Cc3cc(I)c(C)c(I)c3)CC2)=O)cccc([N+](=O)[O-])c1 Cc1cccc(NC(c2nnnn2CC(F)F)C=Cc2ccccc2)c1 N1(C(C=COCC)=O)CCN(C2CCN(C(C34CCC3CC4)=O)CC2)CC1 C(=O)(C(C)(C)C#C)NC1C(C(N(C(C)COCC)CC=C)=O)OCC1 C1(C(=O)NC2(CC(=O)OC)CC2)CCC(C)CN1C(=O)CC(C)F N1(C(CC=C)=O)C2CCC1CN(C(=O)C(C1CCOC1)NC(C)=O)C2 C(=O)(C(C)C(C)S(C)(=O)=O)N(CCN(C(=O)C(C)(C)CF)C(C)C)C CC1CCCCC1(C)C(N1CCC(C(=O)Nc2ccccc2)C(C)C1)=O C1(C(=O)NCCN(C(C(C#C)(C)C)=O)C2CC2)Cc2cc(Cl)ccc2O1 c1(C(=O)NC(C2CN(C(C3CN4CCN3CC4)=O)C2)C)ccc2c(c1)ncn2C C(=O)(CCC1=C(C)NS(=O)(=O)N=C1C)NCC1N(C(C=C(CC)C)=O)CCCC1C c1(CC2(NC(=O)Nc3ccccc3F)CC2)nc(N2CCCCC2)ncc1Cl C(CCC(=O)N1CC(OCCNC(=O)CCc2nccn2C)C1)=C(C)C C1(C(=O)NCC2(C(=O)NCCC=CCCC)CCCO2)CC(=O)CCO1 C(=O)(N=c1cnn(C2CCOC2)[nH]1)c1c(C)occ1 c1(CNC(C2C(CNC(C=CCOCCOC)=O)CCC2)=O)ccc(O)c(C)c1 C1(NC(C2NC(=O)C(F)C2)=O)CC12CCN(C(c1ccc(O)nc1)=O)CC2 Cc1nccc(C(=O)NCC(C)N(C)C(c2cc(C3CC3)cs2)=O)n1 N1(C(N(CCSC)CC)=O)CC2CCC(NC(=O)CC(C)C)C2C1.C1CC1 C(CCCCC(=O)N(CC(C)N(C(=O)Cc1cccc(O)c1)C)C)OC c1(C(=O)NC(C)C(C)(C)NC(=O)CC2C=CS(=O)(=O)C2)ccc2nn[nH]c2c1 c1(C(C(=O)NC2CN(C(C=CC)=O)C(C)CC2)=O)cc(F)c(F)cc1F CC(C)CC(CNC(=O)C(F)CN(C)C)C(=O)NC(CN(C)C)CC(C)C C1(C(=O)NC2CC(C)(C)CN(C(C3C4CC5C(C4)C35)=O)C2)CC2OC(C)(C)OC2C1 c1(C(c2n(C(C)C)nnn2)NCCCn2ccnn2)cnc(N(C)C)cn1 C1(NC(CC2CC(C)N(C(=O)CC3CC4(CC4)CO3)C2)=O)CCOC2(CCC2)C1 N1(C(C(CC)(C)CNC(=O)CCc2cnccn2)=O)CCC(=C(F)F)CC1 Cc1c(C(=O)NCC(C)N(C(=O)CCC2NC(=O)NC2=O)C)ccn1C c1(C(N(CCCNC(C(C)C(F)F)=O)C2CC2)=O)n[nH]c2c1CC(F)(F)CC2 N1(C(Cn2nc(C)c(Br)c2)=O)CC2(CCN2C(=O)C(C2CCCCC2)O)C1 c1(C(=O)NC2(C)CC(NC(c3c(C)cc(C(F)(F)F)s3)=O)C2)ccc([N+](=O)[O-])[nH]1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCCN(C(C2CC2F)=O)CC1c1ccccc1 C1(C(N(C(C)CNC(=O)CC2=CCN(C)CC2)CC)=O)CCCN1S(=N)(=O)N(C)C c1(C(N2CCC(C)C2CNC(C23CCC(C2)C3)=O)=O)cc2n(n1)CCCO2 C1(NC(C(CO)OC)=O)CN(C(=O)C(c2ccccc2F)C)C2CCCC12 CCC(CNC(c1cccc(F)n1)c1nnnn1CCOC)(CC)C(F)(F)F Cc1ccc(C)c(CC(=O)NCCNC(=O)C(c2cccc(Br)c2)C)c1 C12(C(=O)NCC(CN(C(c3c(CC)occ3C)=O)C)O)CCC(CC1)C(C)(C)O2 C1(C)(CNC(C2N(C(C)C)C(=O)CC2)=O)CCN(C(C2CC2C2CC2C)=O)CC1 C(=O)(C1=C(C)NC(=O)NC1CCCSCCN)OCCC N1(C(c2cc(CC)on2)=O)CC2CCC(C(N3CCC(F)(C(N)=O)C3)=O)(C2)C1 n1(CCOC)nc(C)c(C(N2CCCC(C)CC2)C(=O)NC2CC2)c1C C(=O)(CCCCCNC(=O)C(C)(C)C)N1CCC(C(C)O)C1 C12(CNC(=O)NCCN3C(C)CCCC3)CCC(CC1(F)F)C2 c1(CNC(C2CC(C)(NC(CCc3ncn(C)c3)=O)C2)=O)cc(F)ccc1O CCCC(C(=O)NCC1CN(C(C2(C3CC3)CCCO2)=O)C1)c1ccc(Cl)cc1 CC1OC2(C)CC1(C(=O)NCCC1CCN(C(=O)COc3ccccc3)C1)C2 C=C(C)c1cncc(C(C(=O)NCc2cccc(Br)n2)N(CC(C)(C)OC)C)c1 c1(C(=O)NC(C)CCNC(=O)Cn2ncc(Br)n2)cc2c(Cl)cccn2n1 C#CCCCCCC(C(=O)NCC1(CC)CC(F)(F)C1)N(C(C)C(=O)OC)C N1(C(C2(OC)CCSC2)=O)CC2(CCCC(CNC(=O)CCCOC(C)C)O2)C1 N1(C(c2scc(OC)c2)=O)CC(C)(C)CC1CNC(c1cc(C)sc1C)=O c1(C(N2CCN(C(C(CCC)C(C)C)=O)C(C)CC2)=O)cccc2c1C(=O)CC2 N1(C(c2ccn(CCNC(C3C(C(=C)C)OCC3)=O)c2)=O)CCN(C)C(C)(C)C1 CC1(C)CC(=O)NC1SCC1CCC(F)C1 CC(C)CC(O)C(C)C(=O)N1CC2(CC(C(=O)NOCC(O)C(C)C)CO2)C1 C1(CCNC(c2ccc(F)cc2F)=O)CC(F)(F)CN1C(=O)C=Cc1cncs1 N1(C(CC(C)C)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC(C)(C)C1 C(=O)(C#CC1CCOCC1)N(C1CN(C(=O)CCOc2cccc(Cl)c2Cl)C1)C c1(CNC(c2ncn(CC)c2)=O)ncc2ccccn12 C12CCC(CC1)C(=O)NC2.C1(NC(C(C)N(C)C)=O)(CO)CCCCC1 c1(-n2cc(C(=O)OC)nn2)cccc(C(C)(C)NCCN(C)CCC2CCC2)c1 N1(C(CCc2cc(C)no2)=O)CCC2CCC(C1)N2C(=O)C=CCF N1(CC(=O)NCC2CC2(C(F)(F)F)CO)CCNC1=O C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1C)N2C(=O)CC(C)n1ccnc1 c1(C(O)N(C(c2ccc(Cl)cc2)C(N2CCC(CCC)C2)=O)C)ccc(F)cc1 C(C(=O)N(CCC(=O)NC1CC1)C)(C(C)O)NC(c1cnc(OC)s1)=O c1(C(=O)Nc2c(C)nc(-c3ccc(SCCCC)cc3)s2)cc(C)ccc1C C(=O)(C1CCCc2nn[nH]c21)N(C1(CNC(=O)CN2CC3CC3C2)CCCC1)C Cc1scc(C(=O)NCCOC2CN(C(C3(C#N)CCCO3)=O)C2)c1C C1(OC)CN(C(=O)C(c2ccc(F)cc2)SC)CC1NC(=O)C=CCO C1(CC)CC(C(=O)NC2(CCNC(=O)C=Cc3ccncn3)CCCC2)CCO1 C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCN(C(c2ocnc2C(F)F)=O)C1)OC CC(C)C(F)(CNC(=O)CP(C)(C)=O)C(=O)NC1CC(C)(C)OC1=O C1(CNC(c2nc(C3CC3)cs2)=O)CN(C(c2cnoc2)=O)CCCO1 C1(C)(NC(Cc2c(C)occ2)=O)CCCN(C(=O)CC2CCCO2)C1 C(CN=c1cccc(S(=O)(=O)NCCn2ccnn2)[nH]1)N(CCOC)C Cc1nc(C(=O)NCCCCCNC(C2(C)C=CCC2)=O)nn1-c1ccccc1 CC(CNC(=O)Cc1ccc(N(C)C)cc1)CN=c1[nH]cc(C#N)c2ccsc12 C(=O)(CC(O)C(Cl)(Cl)Cl)NC1C(CO)CCN(C(CCC#CC)=O)C1 N1(C(COCCCC#C)=O)CCCC(CCCCNC(C2CCN(C)C2)=O)C1 CCCCC(CC)CCC(=O)NCCC(C)(C)NC(C1CC(=O)NC(=O)N1)=O N1(CCc2cn(NC(=O)Cc3ccsc3CCO)nn2)CC(CO)CC1CO c1(C(=O)NC2CN(C(C(C3CCC(=O)N3)C)=O)CC2F)cc([N+](=O)[O-])ccc1Cl C(N=c1[nH]cnc(Cl)c1F)C12CCC(CNC(=O)C=Cc3cocn3)(CC1)OC2 C1(C(N(C)CC2CCN(C(c3ccn(COC)n3)=O)C2)=O)CC(F)(F)C1(C)C C1(CC(=O)NCCN(C)C(C2(O)CC2)=O)CC(N(C)CCO)C1 C1(C(=O)NC(C)C(=O)NCc2ncc(F)cc2F)CC(C)(C)CCO1 N1(C(C2(F)CCCN(C(C3CCCOC3)=O)C2)=O)CCn2cnnc2C1 Cc1cn2ccc(C(=O)NC3COCC3NC(=O)C(C#N)C(C)C)cc2n1 C(=O)(CC1=CCN(C)CC1)N1C(C(N(CCC(C)O)C)=O)CC(=O)C1 c1(NC(C2(CNC(c3c(OC)ccc(F)c3)=O)CC2)=O)nc2ccc(C)cc2s1 Cc1nccc(C(=O)NCc2ccc(C(=O)NCC(F)(F)C(C)C)o2)c1C C1(C(C(C)NC(=O)CCC2CCOCC2)NC(CN(CCC)C)=O)CCCCC1 C(C(=O)NC1CC(N(C(=O)Cc2ncn(C)c2C)C)C1)(C(C)C)NC(COC)=O C1(C(N(C(C)CNC(c2c(C(F)F)cnn2C)=O)C)=O)CC12CC(C)(C)C2 C=CCC(CC)C(=O)NCC1CN(C)CCN1C(c1cnc(C2CC2)nc1O)=O C=CC(C)(CC)C(=O)N1CC2CC(NC(=O)C(C)Cc3cccc(F)c3)C2C1 C(=O)(C(CNCC(=O)OC)C(C)C)N(CC(N)=O)C(=O)Cn1ccnc1 C1(NC(C(C)Cc2ccco2)=O)COCCN(C(c2cscn2)=O)C1 CN1C(=O)CCCC1C(N1CCCC(C(C)(C)C(=O)NCCCOCCO)C1)=O N1(C(c2c(C)n[nH]c2C)=O)C(C)CC2CN(C(c3ccc4ccnn4c3)=O)CC12 C=CCC(CNC(=O)CC(F)(F)CC)C(=O)NOCC(O)C(C)(C)C c1(C(=O)N(CCCCNC(=O)Cc2nc(C3CC3)cs2)C2CC2)cscc1F c1(C(=O)NC(CNC(C2(CC)CCC2)=O)C2CC2)cccc(C2CC2)n1 c1(NC(c2cc(NC(c3ccc(C)cn3)=O)cn2C)=O)cnc(Cl)c(C)c1 N1(C(C2C(=C)C2)=O)CCOC2(CCN(C(c3cccc(OCC)c3)=O)C2)C1 Cc1cc(C(N2CC(C(O)C(=O)N(CCN3CCOCC3)C(C)C)C2)=O)c(C)nn1 Cc1cc(C(=O)NCCC(C)(C)NC(=O)Cn2cccnc2=O)cc(=O)n1C CC1(C)CN(C(c2cc(C(N)=O)no2)=O)CC1NC(=O)Cn1cnccc1=O c1(C(=O)NC2C(NC(C(c3c(C)noc3C)C)=O)CCCC2)cc2n(c1)CCC2 N1(C(c2c(CC)ncnc2)=O)CC(NC(c2cc3scnc3[nH]2)=O)CC2(CC2)C1 C(=O)(CCN1C(=O)COc2ccccc21)NCC(CC)NC(=O)C(F)C(F)(F)F C=C(C(=O)N1CC2(CC2C(=O)Nc2cc(C)nc(F)c2)C1)C(F)(F)F c1(OC(C)(C)C)cc(Cl)ccc1C(N1CCC(NC(=O)COc2nccs2)C1)=O C=CC(CC)CC(=O)NC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)C1C(CC)C1 Cc1nc(Br)ccc1NC(=O)C(N1CCC(CNC(C2CCCCC2)=O)C1)=O C1(NC(CCN(C)CC)=O)CN(C(c2cc(Cl)cnn2)=O)C2(CCCOC2)C1 C1(C(=O)OCC)CCN(C(=O)N(c2cccc(OC)n2)C)C2COCC12 c1(CN2C(C(=O)Nc3c(C)nccn3)CC2)c[nH]c2cccc(C)c12 c1(SC)cc(C)c(C(=O)NC(C2CCN(C(=O)Cc3cn[nH]c3)C2)C)o1 c1(C(=O)NCC2(CCNC(C(C)SCCCC)=O)CC2)ncc(F)cc1C N1(C(C(F)=C(C)C)=O)CC(F)(F)CC1CCNC(c1ncoc1C1CC1)=O Cc1ccc(OCCCNCc2ccncc2-c2cnc(F)nc2)c(F)c1 C1(O)(CCNC(CC2(NC(C)=O)CC2)=O)CCCN(C(c2ccon2)=O)C1 Cc1nc(C(=O)NC2CC(F)CN(C(C3CCC(O)CC3)=O)C2)c2n1CCCC2 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(OC)C(NC(c2cc(Cl)n(C)n2)=O)CC1 c1(OC)ccc(F)c(C(C(=O)NCc2ccco2)N(C2CCSC2)C)n1 c1(NC(C2CN(Cc3c(O)cc(Br)cc3F)CC2O)=O)cc(Cl)c(Br)cc1Cl N1(C(C2N(C(CCC)=O)CSC2)=O)CCC(C)(CNC(C2CNC(=O)N2)=O)CC1 C#CC1(NC(C2(CNC(=O)C(O)CCSC)CC3(CC3)C2)=O)CCC(C)CC1 N1(C(c2c(OC)csc2)=O)CCOCC1C(=O)NCC(C)C(C)(C)C c1(C(=O)NCCN(c2nnc(CO)s2)CC)c(C)oc(C)c1C C1(CN2CCC(N(C(=O)C(c3ccccc3)C3CC3)CC)C2)CC2CCCC2C1 c1(C(N2CCC(N(C(CCC#C)=O)C)C2)=O)nc(C(F)(F)F)oc1Br c1(C(=O)NCC(C(C)C)NC(=O)CCC2CC2)cccc2occ(Br)c12 C12NC(=O)N(CCN3CCSCC3=O)C(CF)=C1C(=O)n1cc2cn1.CC C1(CC(=O)NCC(CNC(c2c(C(N)=O)coc2)=O)(C)F)CCCCC1O N1(C(C(c2c(C)noc2C)C)=O)CC2CC(NC(=O)CCC3CCC3)C1C2 Cc1ccccc1C=CC(=O)NC1CC1C(=O)Nc1cncnc1 CC1CC(C(=O)NC2CC23CCCC3)CN1C(=O)COC1CCCCCC1 n1(CC(=O)NCCN(CCC)C(C2CC2C(C)(C)O)=O)ncn(C)c1=O C1(C)(C(=O)NCC(C2CCCC2)NC(CN(c2ccccn2)C)=O)CC1(F)F C1(CNC(C2(OC)CCSC2)=O)COC(C)(C)CN1C(=O)COC1CCC1 c1(SC)nccnc1C(F)(F)F.C1(C(=O)NC23CN(C2)C3=O)(CC)CC1(F)F Cc1ncc(C=CC(=O)NCC2(C)CC(NC(C3CC=CCO3)=O)C2)s1 N1(CCO)CCCCC1c1cccc(O)c1.C(=O)(C(C)NS(C)(=O)=O)N(C)CCO CC(C)CS(=O)(=O)NC1CC2(CCO2)C1 C1(CC(N2CCC(C(C)NC(c3cnco3)=O)C2)=O)CCCC(F)(F)C1 Cn1cnc(C=CC(N2CCC(C(F)CNC(c3cc(F)c[nH]3)=O)CC2)=O)c1 Cn1nc(CNC(=O)CC2CCCCO2)cc1C(N1CCC(C)(C)C1)=O C=C(C)CC(C(=O)NC1CC2CC(NC(c3nc(=O)n(C)[nH]3)=O)C2C1)NC(C)=O N1(c2n(CC(C)C)c(C(c3ccccc3Br)O)nn2)CC2(C1)CC(C)(O)C2 C1(C(N2CCOC(C)C2C)C(=O)NCC2CC2)CCC2COCCC2C1 C1(C(=O)Nc2cnn(C(F)F)c2)COCCN1CC1CC1(Cl)Cl C(CNC(c1ccc(C(N)=O)c(Cl)n1)=O)(CCS(C)(=O)=O)OC CC1CN(C(c2ccnc(CC(C)C)n2)=O)CCC1N(C(=O)C(=O)NC1CC1)C C1(OCC)CC2(C1)CC(NC1CN(C(=O)CC(C)(C)SC)C1)C2 C1(F)(CNC(c2cnccn2)=O)CC(NC(C2CCC3CC23)=O)C1 C1(C(C)C)CN(C(C2CCCCS2)=O)CCN1C(=O)CC1CCC(C)CC1 c1(-c2cc(C(=O)NC(C)CNC(C3CCCS3)=O)sn2)ccc(Cl)cc1 C1(NC(CCOCCOC)=O)CC2(CCN(C(c3cc(Cl)ccc3C)=O)C2)C1 c1(OC)ccccc1OCC1(C(N2CC3C(CN)(C3)C2)=O)CC1.C1C(=O)N1.N(C)C c1(C(=O)NCC2(OC)CN(C(=O)CC(C)SC)C2)nc(Cl)sc1Br C=C(Cl)C(C)(C)C(=O)NCC(O)CN(C(=O)COCC(=O)OCCCC)C C1(O)(CNc2c(C)cc(C)o2)CCCN(C(=O)CCOc2cccc(F)c2)C1 CN1CCCC(C(N2CCCC2C(C)(C)C(=O)NCCC2CCCOC2)=O)C1 C1(NC(=O)CC(F)(F)F)CN(C(=O)C=Cc2cccc(Cl)c2)CC2CCCC12 c1(SCC)ccc(C(N2CC(OC)CC2CNC(C2CCC(=O)N2)=O)=O)cn1 c1(CCC)n[nH]cc1C(=O)NCC(CC)NC(=O)CC(C)N(C)C C1(C(=O)NCC(C)(C)NC(=O)C(F)=C2CCC2)CCCN1C=O C(CS(=O)(=O)C(C)(C)C)N(C(=O)Nc1ccc(C(CC)C)cc1)CC C1(CNC(COC)COC)CCCC(CNC(c2cccc(CO)c2)=O)C1 C1(c2nnnn2C2CC(F)(F)C2)(NC(c2cccc(Cl)c2)C)CCCC2(CC2)C1 c1(C(=O)NCCCN2CCC(NC(C(C)CF)=O)C2)n[nH]c2ccc(Cl)cc12 C(=O)(C(CC(F)F)NC(C1CC(C)(C)C1)=O)NC1(C)CS(=O)(=O)C1 Cc1ccc2c(c1)CCN2C(C1OCCC1(C)C)C(=O)NC1CCCC1 C1(CC(=O)NCC=CCNC(=O)CCc2nc(C(F)(F)F)n[nH]2)CC2CCC1O2 C1(C(N(C2CC2)CC)=O)CCCN(C(=O)C#N)C1 C1(C(N2CCC(=C)CC2)=O)CN(C(=O)C(C)NC=O)CC(C)(C)C1 N1(C(CC(=C)Br)=O)CC(CNC(=O)CCCNC(N)=O)C2(CCC2)C1 c1(C(=O)OC)cnccc1N1CC2C(CNC(c3nccnc3C)=O)C2C1 N1(C(=O)CCOCC(F)F)CC2CC1CN2C(c1nccc(Br)c1O)=O N1(C(c2nc(C)sc2)C(=O)NC2CCOCC2)CCCC2NC(=O)CCC12 c1(C(=O)NC(C2(CNC(C3C(C)C3)=O)CC2)C)ccc(Cl)c2ccccc12 N1(C(C(C(C)C)(C)O)=O)CC2C3CCC(C2C1)N(C(=O)Cc1cccc(F)c1)C3 C1(CNC(C2CC3CCC2O3)=O)CN(C(C2CCS2(=O)=O)=O)CCCO1 C(c1ccc(C(N)=O)o1)=CC(=O)NCC(C)CNC(C1CCO1)=O C1(CN(C(c2c(OC)n[nH]c2)=O)C)CC(F)CN1C(c1cc(OC)n(C)n1)=O CCC(C)(C)CC(=O)NC(C)C(C)NC(c1ncoc1-c1cnn(C)c1)=O C1(C(=O)NCc2n(CC)ncn2)CCCCN(C(c2ccc(CO)cc2F)=O)C1 N1(C(C2C(C)CC(=O)CC2)=O)CCCC(CNC(c2cncc(Cl)c2)=O)CC1 c1(C(N2CCC(C)(CNC(=O)C(F)C(F)(F)F)CC2)=O)cc2c(nc1N)CCC2 N1(C(COCc2c(C)ncs2)=O)CCOC(C(C)NC(=O)CSC(=N)N)C1 C1(NC(CSCC=C)=O)CCCN(C(=O)CCCOC(C)CN(C)C)C1C N1(C(Cc2nnn(C(C)(C)C)n2)=O)CC(NC(C23CCCC2C3)=O)CC(O)C1 N1(C(CC(=C)C)=O)CCC2(CCN(C(=O)C(C)C(F)F)CC2)C1 C#CC1CCN(C(=O)OC(C)(C)C)C1.c12nc(C)c(s1)CN2C N1(C(c2c(C)nco2)=O)CC2(C1)SCCC2NC(c1cnc(O)n1C)=O Cc1ccc(O)c(NC(c2cnc(C)cn2)=O)n1 c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)C2)C)ccc(CO)cn1 Cc1oc2ccccc2c1C(C)NCCn1cc(C2(S(=O)(=O)N(C)C)CC2)nn1 N1(C(C2CC=C(C)CC2)=O)CCC(C2CC2)(CNC(=O)Cc2ccnc(C)c2)C1 c1(C(=O)NCCn2cc(CCC3CCOCC3)nn2)ncc2ccccn12 C1(C(=O)NC2CC(CNC(=O)C3=CCCOC3)C2)CCn2c(O)nnc2C1 N1(C(C2(C)N(C(c3nc(C)sc3C)=O)CC=C2)=O)CCC2(CC(CO)C2)C1 c1(OC)ccc(-c2cnc(C(=O)N(CC#N)C3CC3)cc2C)c(C)n1.C(=O)N N1(C(C2C(C)(C(F)F)C2)=O)CC(CNC(c2cnoc2C2CC2)=O)C2(CCC2)C1 O=S(=O)(c1cc2cc(F)ccc2o1)NCCn1cc(C2(O)CC3CCC2C3)nn1 N1(C(c2c(CC)ccs2)C(=O)NC(C)CC)CCC(C2(O)CCC2)CC1 c1(C(N2CC(CNC(C=C(C)C(F)F)=O)OCC2)=O)cc(N)cnc1Br CC1CCC(O)(CNC(C2CCC(NC(C3CC4(CC4)CN3C)=O)C2)=O)C1 c1(C(N2CCC(N(C(CCCCCCC)=O)CC)C2)=O)noc2ccc(F)cc12 C1(CCNC(CNC(=O)OCC=C)=O)C(C)CCCN1C(=O)Cc1sccc1C C1(NC(C23OCC(CC)(C2)C3)=O)CC2(C1)CC(NC(c1ccccn1)=O)C2 CCCCCC(=O)N(C)CCN(C(=O)C(C(=O)OC(C)(C)CC)OCC)C c1(N2C3CC(=C)CC2CCC3)nc(=NCSC2(OCC)CC2)[nH]c2c(F)cccc12 CC1COC(C)(C)CN1C(Cc1ccccc1)C(=O)N(C)C CN1CCOC(C(=O)NCC2CCCCC2NC(=O)C=Cc2ccc(C)o2)C1 c1(C2(C(=O)NC(C3(O)CN(C(=O)C(O)CO)C3)C)CCC2)ccc(F)c(Cl)c1 Cc1[nH][nH]c(=NC(=O)C2CCC2NCc2ccc3n[nH]cc3c2)c1Br C1(CNC(c2cccc(CC)c2)=O)C(C)CCCN1C(=O)CCC1CCC1 N1(OCC)CCC(C(=O)NCCOC(C)C)CC1.C12(CC1)CS2 C1(C(NOCCC(C)C)=O)CN(C(=O)CCc2cccnc2)CCC1(C)C C1(CNC(=O)CCC2CCCC(=O)N2)(CO)CCN(C(c2cc(Cl)n[nH]2)=O)CC1 CC(C)(C#CC(=O)NC(CC#N)c1ccco1)CNC(C1CC1F)=O C1(NC(CC2N(C(C(N3CCOC3=O)C)=O)CC2)=O)CC2(CCCC2)C1 c1(OCC(=O)O)ncccc1CNc1cccc(C(N2CCOC(O)C2)=O)c1 c1(C(N2C(CCCNC(C3C(CC)OCC3)=O)CCC2)=O)ccccc1Cl c1(NC(=O)Nc2cc(OC)c(OC(F)F)cc2)ccc(S(C)=O)cc1.C1CO1 Cc1nccc(C(=O)NCC23CC(NC(c4cc(C(C)C)oc4C)=O)(C2)C3)c1C N1(CCCC)CCCCC1CCNC(=O)CC1CCC(C)O1.N12CSCC1C2=O C1(CCC)CN(C(c2cccc(COC)c2)=O)CCN1C(=O)C(C)C(F)F c1(O)cccc(NC(=O)C(CC)NCCCCCC)c1 c1(CN(C(C#C)C)Cc2cccs2)ccc(OC)c(-c2ccnc(C)c2C)c1 C1(=O)CCO1.C(C(=O)NC)OCCOCC N1(C(C(N2CCOCC2)C)=O)C2CCC1C(NC(=O)COC1CCC1)C2 C(=O)(C1=CCCNCCC1)N(c1ccc(F)cc1)CC#N C(C)(C)(CCCCC(=O)N1CC2CC(NC(C34CCC3CC4)=O)CC2C1)OC c1(C(=O)NC2CC(C)N(c3cc(C4CC4)ncn3)CC2)occ2c1CCOC2 N1(C(C2CCCC(=O)N2)=O)CC2(CCC2NC(=O)C(=C2CCCCC2)F)C1 N1(C(CC(CC)(F)F)=O)CCOCC12COCCN(C(=O)CCC(C)O)C2 C1(NC(C(=Cc2ccco2)C)=O)CCN(C(C2CN(C)CCO2)=O)CCC1(F)F c1(C(=O)NCC(C)NC(c2nnn(COCC)c2N)=O)ccc2c(c1)CN(C)C2 CN1C(=O)CCC1(C)CNC(C1CN(C(c2ncncc2N)=O)CC12CC2)=O N1(C(CCCC(=O)NCC)=O)CCC2(CC1)CC2CNC(=O)C(C)n1cncn1 O=C(C1=CC2(CCN(C(c3cccc(=O)o3)=O)C2)C1)NCC(c1ccccc1)O N1(C(=O)COCCN2CCOC2=O)CCC(CO)C1c1ccccc1 Cc1ncc(Cl)cc1CC(N1CCC(NC(=O)CC2CNC(=O)C2)C(O)C1)=O c1(NC(C(CN(C)C)NC(c2n(CC)c(O)nc2)=O)=O)c(C)cc(C)cc1C c1(CC(N2CC(CCNC(=O)C=Cc3cn[nH]c3)OCC2)=O)cc(F)ccc1O c1(CN2CCCC(C(=O)Nc3c(C(C)=O)con3)C2)cnc2c(Br)cccc2c1 Cc1cc(C(=O)NCCC2(NC(=O)CCC3CCC(=O)N3)CCC2)c(C)cc1Cl c1(C(=O)NC2C(CNC(C(C)n3ccnc3)=O)COC2)ccc(P(C)(C)=O)o1 C1(C(=O)NCC2(F)CC(CNC(C(C)CN3CCOCC3)=O)C2)CCCS1(=O)=O CC1(C(=O)NCCC2(CNC(c3cncnc3)=O)CC2)CCC(F)(F)C1 C1(C(=O)NCC(c2ccccc2)NC(=O)CCS(C)=O)(NC(C)=O)CCCCC1 C(=O)(C1=CCCOCC1)N1CCC(CC)C1CNC(c1c[nH]c2nccc-2c1)=O N1(C(C2C(C(=O)OCC)CCCC2)=O)CC(NC(C23CCC(C2)C3)=O)C(C)(C)C1 CC1CC(N=c2ccnc(NCc3ccc(N)cn3)[nH]2)CCO1 c1(OC)cccnc1C(N1CCOC(CCNC(=O)C(C)NC(N)=O)C1)=O Cc1ccc2c(c1C(=O)O)CCCN2C(C1CCC(=O)N1C1CC1)=O c1(N2CCC(NC(c3cc(C)c(C)[nH]3)=O)C(C)C2)nc2ccc(N)cc2s1 c1(C(=O)NCC23C(CN(C(C4ON=C(CC)C4)=O)C2)C3)sccc1S(N)(=O)=O C1(C(=O)OCC)CC2CC1CC2NC(c1ncncc1C)=O.C12CC(C1)NC2=O c1(CC)nccnc1N(C)CC1CCN(C(C2CN(C(C)=O)C2)=O)C1 c1(NC(COC)=O)ccc(C(=O)NCCNC(=O)CS(C)(=O)=O)cc1.OCC N1(C(CC(C)N2CCCC2=O)=O)CCN(C(=O)COCC(F)(F)F)CC12CC2 c1(C(=O)NCC(C)CN(C)C(C2CC(F)(CO)C2)=O)ccc2nn[nH]c2c1 c1(CC(=O)N(C(c2cccc(OC)c2)CNC(C)C)CC)cnc(Cl)c(F)c1 N1(C(c2c(NC)cc(Cl)cc2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)CO)C2 N1(C(CCC=C=C)=O)CCC(C(N2CCC(n3ccnc3)C2)=O)CC1(C)C c1(OCC(=O)NCCC2CCN(C(c3cnc(C(C)C)o3)=O)C2)ccc(F)nc1 N1(C(CC(CC)SC)=O)C2CCC(C2)C1C(N1CC(=O)NC(=O)C1)=O O=C(C#CC1CCCOC1)NCCC1CN(c2ncnc(Cl)c2F)C1 CC1CCCCCC1NC(C1OC(C)(C)OC1CNC(=O)OC(C)(C)C)=O C1(COC)CN(C(=O)C(c2cc(Br)co2)=O)CCN1C(=O)CCn1cncn1 c1(CCC(C)C)n[nH]c(=NCC2CC(NC(c3ccc(NC(N)=O)cc3)=O)C2)o1 C1(C(=O)NCC(CC)N(C)C(c2cc(CO)ccn2)=O)CC=CCC1C C1(C(=O)NCCCN(C(c2cc(C(C)C)c(O)cc2)=O)C)COC2(CCC2)CO1 c1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)cc(C)ccc1N N1(C(C2C(C)C2)=O)CC2CN(C(=O)C(C)(C)C(F)(F)F)CCC12 N1(C(c2c(C)cncc2F)=O)CCC(C)C(C)(C)C1 N1(C(C(CC)C)=O)CCN(C(=O)CCc2nc(C(C)SC)no2)C(CO)C1 C(=O)(C1=NOC2(CCC2)C1)NC(C)(C)CNC(=O)CCCc1ccccc1Cl c1(OC(C)C)nn(-c2ccccc2)cc1C(N1CCCC1C(O)C(F)(F)F)=O Cc1cc(=O)ccn1CC(=O)NCCC1CN(C(=O)CC2(O)CCC2)CCO1 O=C(CCCCC1CC1)NCC1(F)CN(C(c2c[nH]nc2F)=O)C1 c1(C(=O)NC2CC(CO)N(C(=O)Cc3cc(Cl)ccc3Cl)C2)csc2nnsc12 C1(CC(=O)NCC2C(NC(C3(CC)CC(C)(C)C3)=O)CCC2)CCCCC1(F)F C1(C(=O)NC(C)CN(C)C(c2ccc(F)c(Br)c2)=O)CC12CCC(F)(F)CC2 CCCC(C(=O)N1CCCC(CN(C(C2CC2(C)C)=O)CC)C1)NC(C)=O C(C1=CCN(C(=O)C(C2CCCN(C)C2)(C)C)CC1)NC(c1c(C)noc1Cl)=O c1(C(=O)NC2(C)CC(NC(C3COCCC3(F)F)=O)C2)ccc(=N)[nH]c1Cl N#Cc1ccc(C(=O)NCC(F)CNC(c2cc3c(s2)CCC3)=O)c(F)c1 C(=O)(CCS(C)(=O)=O)N1C(CNC(CNC(C(CCC)C)=O)=O)CC1 C1(C(C)NC2CC3CC2CN3)CCCC(C)(C)CC1 C1(CNC(CCC(=C)Br)=O)CCN(C(c2nocc2C(=O)OC)=O)CC1C N1(C=O)CC(C(=O)O)C2(C1)CN(C(=O)C=C(C)C)C2.c1(OC)ccc(C(=O)OC)c(I)c1 N1(C(C2C(CCC)C2)=O)CC2(C)CC1(C(=O)N(C(CC)CC)C1CC1)C2 Cc1oc(CO)cc1C(=O)NC1(CC(=O)NC2CCN(CCCO)C2)CC1 N1(C(C=C(C)Cl)=O)CCCCC(NC(c2cc(Cl)c(Cl)cc2N)=O)CC1 C1(CNC(N2C(C)CC(C(=O)OC)C2)=O)CCCCCC1C1CC1 c1(C2(NC(C(n3cc(C(CC)OC)nn3)C)=O)CC2)cc(Cl)ccc1C c1(CNC(N2CCOC3CC23)=O)ccc2ccccc2c1Br N1(C(C(CCSC)O)=O)C2CCC1C(CNC(c1oc(CC(C)C)nc1C)=O)C2 c1(OC)cncc(C(=O)NC2COCC2NC(=O)CSc2c(C)n[nH]c2C)c1C C1(NC(C2CC(C)NC(=O)C2)=O)CN(C(=O)C(C)(C)c2ncco2)CC12CCC2 C12CC3CC(CC13)NC(=O)CO2.c1(OCC=CC(CCCOC)=O)ccccc1 c1(C(=O)NCC2C3CN(C(C4CC(C)OC4)=O)CC32)c(Cl)nc2ccccn12 CCC(C(=O)NCC1(OC)CCN(C(c2ccc(F)c(F)c2)=O)C1)C(C)(C)CC C1(C2CCCN(C(C3(C)CC3(F)Cl)=O)C2)(NC(C(COC)(C)C)=O)CC1 Cc1cc(-c2nccnc2C(N2CC(=O)NC(C)C2)=O)ccc1C#N C1(NC(COCCC=C)=O)CC12CCN(C(c1sccc1OC)=O)CC2 N1(C(c2ccc(OC)c(Cl)n2)=O)CCC2(C1)CN(C(c1ocnc1C)=O)C2 C1(CC=C)(C(=O)NCC2(NCC)CCC2)CCCN1C(=O)C(CCOC)OC n1(CC(=O)NCC(C)CNC(C2(C)CC3CCC2O3)=O)ccc2ccc(F)cc12 C1(NC(C(C)NC(=O)C(N2CCOCC2)C)=O)C2CCCC1COC2 C(CC(C)CC(C)(C)C)NC(Cn1cc(CNC(c2ccc(C)c(C)c2)=O)nn1)=O c1(C(=O)NC2CC(N(C(Cc3c(C)cnn3C)=O)C)C2)nc(C)[nH]c2nccc1-2 C(C(C)(C)C(=O)NCC1CC(O)CN1C(c1ccccc1Br)=O)N(C)C N1(C(C2CC(CC(C)C)C2)=O)CCCC2(C1)CN(C(=O)Cc1ccsc1)CCO2 C=C(C)C(C)(C)C(=O)NC1C2CC(NC(C3CCC(F)C3)=O)CC12 c1(C(N2CC(CNC(C3CC(=C)C3)=O)C3C2C3)=O)cc(Br)cc2ccccc12 CCC(C(=O)NCCCC1N(C(C23CC(CF)(CO2)C3)=O)CCC1)C(C)(F)F c1(C(=O)NCCc2ccc(C(N3CC(C(C)C)C3)=O)cc2)cc(Br)cnc1O N1(C(C(OC)OC)=O)Cc2occ(C(N3CCC(C(C)CO)C3)=O)c2C1 c1(C2C(NC(C3C(NC(CNC(=O)NC)=O)C3)=O)C2)cncc2ccccc12 CC(C)CC(C)C(=O)NCC(C)(C)C(=O)N(C(C)CN(C)C1CC1)C N1(C(C#CC)=O)CCN(Cc2cncc(C)n2)C(CN2CCOCC2)C1 c1(CC(=O)N(CCN(C(C2C(=C)C2)=O)CC)CC)c(C)cnn1C c1(OC)cc(C(=O)NCC2CC2NC(C23CC2COC3(C)C)=O)cc(C)n1 c1(N(CC(C)NC(C2CS(=O)(=O)CC(=O)N2)=O)C)ncc([N+](=O)[O-])cc1Cl C1(NC(=O)NC2CCCC2)CCCN(CCO)C1.c12nnnn1CCS2 c1(C(=O)NC2(C(=O)NCC3(O)CCC(C)C3)CCSC2)cc(N)cc(F)c1 Cc1cc(F)cc(C(=O)NCC2CCCN(C(c3cc(C(F)F)on3)=O)C2)c1N C1(F)(C(=O)NCC=CC(=O)NC(C2CCCO2)CO)CCCCC1 CC(F)(F)CCC(=O)N1CC2C(CNC(C3(C(F)(F)F)CCCCO3)=O)C2C1 C(CCC(C)C(=O)NCC=CC(N1CC(=O)NCC1C)=O)OC c1(CNC(CCCC)=O)ccc(CNC(=O)CC2CCC(=O)N2)c(F)c1 CCC(CC)C(C(=O)NC1CC(O)(CNC(=O)CC2C(C)(C)C2(C)C)C1)OC CC1=C(C(=O)NC2CCN(C(=O)C=CC3CCCO3)C2(C)C)CCC1 c1(C(C)C(=O)NCCC2CCN(C(C3CN(C)C3)=O)CC2)noc2ccccc12 Cc1cn(CC(=O)NC2CC2CNC(c2nnsc2C2CC2)=O)c2ccccc12 C1(NC(CCCOCCC)=O)CCCN(C(c2ccc(C)c(C)c2)=O)C1C c1(CC)oc(C)cc1C(=O)N(C(CNC(c1cnc(O)n1C)=O)C1CC1)C CC1SCCN(C(c2cc(C(=O)NC3OC4CCC3C4)nn2C)=O)C1C C1(NC(C(CC)C)=O)CC1C1CCN(C(c2cc(NC(C)=O)ccc2F)=O)CC1 C(=O)(C(C)(C)CC1CC1)N(CCCCN(C(=O)CC1CC1(Cl)Cl)C)C Cc1nccc(C(N2CCN(Cc3ccccc3)CC2C)=O)c1O O=C(CCCCO)Nc1cccc(C(N2CCC(NC(C3CC3F)=O)CC2)=O)c1 C1(C)(CNC(c2cc(SC)oc2)=O)CCN(C(=O)CCC2CCCOC2)C1 C(=O)(C(C)CC(C)CC)NCC(COC)NC(c1cccc(OC(F)F)c1)=O C(CC(C)C)(C(=O)N(CC(C)NC(=O)CCc1ncccc1C)CC)OC C=CCC(CNC(=O)CC1COCCO1)C(=O)N(C)CC1CC1 c1(C(c2nnnn2C)Nc2cccc(OCCCOC)c2)ccc2cc[nH]c2c1 C(C(=O)N(C1CCCCC1)CC=C)(C(C)C(C)(C)C)N1CCC(O)(CC#C)CC1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(N=[N+]=[N-])CC1C(=O)NC(C1CCCC1)CO c1(OCC)ccc(C(N2CCC(N(C)C(c3ccc(C)cc3Br)=O)C2)=O)cc1O C(=O)(C1=C(Cl)CCC1)NC1CCC(NC(=O)CC2CC3CC3C2)C1 C1(CNC(C2C(C(C)C)C2)=O)CN(C(=O)CCC=Cc2ccccc2)CCCO1 c1(C(N2CCN(C(C(CC(C)C)F)=O)CC2)=O)ccc2c(c1)NS(=O)(=O)C2 CC(C)CC(C(=O)NCC(C)CNC(C1CC=CC1)=O)N1CCCC1=O N1(C(C(Br)=C(C)C)=O)CCN(C(=O)CCS(C)=O)CC(O)C1 c1(C(=O)NC2CC(NC(C3OCCC(C)(C)C3)=O)C2)ccc2ccccc2c1 Cc1cccc(Cl)c1C(=O)NCCOCCN(C)C(c1nscc1N)=O Cc1[nH]nc(CNC(=O)C=CCNC(=O)CC2CCCCO2)c1C N1(C(C2(CC#C)CCCO2)=O)CCCC(N(C(=O)C=CC=C(Cl)Cl)CCO)C1 c1(C(=O)NC(C2(O)CN(C(c3cc(SC)c(C)o3)=O)C2)C)cnn2c1N(C)CC2 C(CN=c1[nH]nc(C2CC2)s1)C1C(C)CN(C(=O)CCOCC(F)F)CC1 C1(C(=O)OC)CN(C(=O)CNC(=O)CC(C)C)CC1C N1(C(C(C2CC2)OCC)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)CC1C C1(CNC(C=C(C)C2CCC2)=O)CCN(C(=O)CC2CCOC2)CCC1(F)F C1(CC(=O)NCC(CNC(c2ccn(C3CC3(F)F)n2)=O)OC)CCC(C)(C)C1 CC1c2c[nH]nc2CCC1C(N1CC(CNC(c2ccc(C#N)nc2O)=O)C1)=O Cc1cccc2nc(C(=O)N(C)CCN(C(=O)CCn3ccccc3=O)C)cn12 Cc1noc(C(=O)NCCCCCNC(=O)C(F)(F)c2csc(C)c2)n1 C(=O)(C#CC1(C2(C(=O)OC(CCC)C3CC3)CC2)COC1)OC(C)(C)C C=CCC(CNC(C1CC(C)N(C)C1)=O)C(=O)N1CCC(C)(CO)C1 C1(C(=O)NC2CC(O)(c3ccncc3)C2)CCCC2(CC2)C1 C1(C(C)C)CCC(C)CC1C(=O)NC1CCN(c2nc(-c3ccccc3)ns2)CC1 C1(NC(c2ccn(COC)n2)=O)CN(C(c2ccc[nH]2)=O)CC1n1ccnn1 C(C(C)(O)CNCC)NC(=O)OC(C)(C)C.CCC(CN)O CC1CCN(C(c2sccc2C#N)=O)CC1NC(c1c(Cl)cnn1C)=O c1(C(N2CC(C#C)(C(=O)NCCP(C)(C)=O)C2)=O)ccn(C)c(=O)c1 C1(F)(CNC(C2CCCO2)=O)CCN(C(c2cccc(-c3ccoc3)c2)=O)C1 C1(CCC(=O)NCC(C=C)(C)C)CCCCN1C(C1C(C)(C)C1(F)F)=O C1(C(N(CCOCC)CC)=O)CCN(C(=O)CC2CCCC(=O)N2)CCO1 CC1=NNC(=O)C1CC(N1CCOC(CNC(C23CC(C(F)F)(CO2)C3)=O)C1)=O Cc1cc(Cl)c(C(=O)OCC(N2CCS(=O)CC2c2cnn(C)c2)=O)cc1C CN1CCOC(C(=O)N(C)CCOCCNC(c2cnn(C)c(=O)c2)=O)C1=O C(=O)(CC(C)CC(=O)NCC1CC1CNC(c1cc(C(F)(F)F)no1)=O)OC c1(C(N2CC3(CN(C(CC(C)OC)=O)C3)C2)=O)cc(Br)cc2c1CCN2 CC(C)CCCCCC(=O)N1CC2CCC2(CCNC(c2ncc(F)cn2)=O)C1 N1(C(c2c(CC)csc2)=O)CCCC1(C)CNC(=O)C=CCN(CC)CC c1(OCC(C)N(Cc2ccccc2)NS(=O)(=O)CCOC)ccccc1Br C1(NC(c2ccc(CC)nc2)=O)CCC2(C1)CN(C(=O)C(C)(C)Br)C2 c1(COCCCC(C)C)cccc(-c2ccccc2)c1F.C1C(C)NC(=O)N1 c1(C(=O)N(C(C(CCCN2CC=C(C)CC2)OC)=O)C2CC2)ccnc(F)c1F C=CCC(CC)C(=O)N1CCC(CCNC(c2cccc(CC(F)(F)F)c2)=O)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCN(CC(=O)N(C(CC(C)C)C)C)CC1 N1(C(c2scc(C)c2)=O)CC2CCOC2(CNC(=O)C(O)C2CC2)C1 S(=O)(=O)(c1ccc(NCCF)c(Cl)c1)NC(c1cc(C)no1)C CCC(CC(=O)NCC1CC(NC(=O)CCc2ccsc2Cl)C1)C(C)C CC1CN(C(C2CCCSC2)=O)CCCN1C(C1(CO)CC1)=O C(CCCNC(C)(C)CN1CCCC1)C1(OC)CC1.C12(CC1)CC(=O)N2 C1(NC(c2cn(CC)nn2)=O)CC2CCC(C1)N2C(C1CC(OC2CC2)C1)=O Cc1cccc(C(=O)NC2COCC2NC(=O)C(C)(O)C(C)C)c1Cl C1(NC(COCC)=O)CCCC12CN(C(=O)CCn1ccnc1)C2 C1(NC(c2cn(C)nn2)=O)CC2CC(C1)N(C(c1ccccn1)=O)C2 C(=O)(C1=Cc2ccccc2C1)NCCCCC(=O)Nc1c(OC)noc1C c1(N(C)C)ccc(C(=O)NCC(C2CCOC2)O)cc1 C(=O)(CCCCC1CC1)N1CC(CC=C)(C(=O)NCC2(C(N)=O)CCCC2)C1 N1(C(C2(C(C)C)CCN(C(C=C(C)C(C)C)=O)C2)=O)CC2CC(O)CC1C2 c1(C(N2CCCCC(N(C)C(c3ccsc3)=O)C2)=O)c[nH]c(=O)c2ccnn12 c1(C(=O)NC(CNC(c2nc(CC)sc2)=O)CC(C)C)cn(C)c(=O)cn1 Nc1ccc(F)c(C(N2CCN(C(=O)CN3CCS(=O)(=O)CC3)C3CC23)=O)c1 C(=O)(CCCNC(=O)C(C1CCCCC1)NC(=O)C(n1ccnc1C)C)NC C1(C)(OCC(=O)N(CCC(=O)NCC#C)C)CN(C(=O)C(C)NC(N)=O)C1 c1(OC)cc(C2(N(C)C)CCOCC2)ccc1CN1CCC(c2ccc(C)cc2)C1 Cc1cc(C(=O)NC(C)CNC(c2csc(Cc3ccccc3)c2)=O)nc(O)c1 c1(OC)cc(OC)nc(C(=O)NCC2(C)CCN(C(C3NC(=O)CC3C)=O)C2)n1 Cc1ccc(Cl)c(C(=O)NCC(c2ccc(F)cc2)NC(c2csnc2C)=O)c1 c1(C(=O)NCCC2(O)CCCN(C(=O)CC(F)(F)F)C2)cnnc2ccccc12 c1(C(=O)NC2C3CN(C(c4c(C)nc(Br)o4)=O)C2C3)ccc2c(c1)C=CCC2 c1(C(N2CCCC(NC(C3C(=C)C3)=O)C2)=O)cc(Cl)cc(Cl)c1F c1(C(=O)NCC2CCN(C(C=C(CC)C)=O)C2)ccc(OC)c(-n2cnnn2)c1 N1(C(=O)C(F)F)CCOC2(CCCN(c3ncc4c(Br)cccc4n3)C2)C1 c1(C(=O)NC(C(=O)NC2CCC(=O)NC2=O)CC2CCC2)ccn2ccnc2c1 C1(CNC(C=CCCC(C)C)=O)CN(C(C2(F)CCC2)=O)CCC1C(F)(F)F CC1(C)CC(NC(=O)CCCCc2ccccc2)CN1C(=O)C1=CCCOC1 C(=O)(C(CC)CCc1ccccc1)N1CCC(CC=C)(NC(C2CC2CC)=O)C1 N1(C(C(C)Sc2ccc(F)cc2)=O)CC(NC(c2ccnc(Cl)c2)=O)C(C)C1 CC1(C)CC(C(N2CCC(C(=O)NCC3CCCC(=O)N3)CC2)=O)CCO1 N1(C(C(C)SCC)=O)CC(C(N2CCCC(F)(F)C2)=O)C2(CC2)C1 C(CC(=O)Nc1cncc(C)c1)(CC(C)C)NC(C12CCC(OC)C1C2)=O C(c1cccc2ccccc12)=CC(N1CCCCC(NC(=O)C=CC2CC2)C1)=O N1(Cc2cn(C3C(OC)CCC3)nn2)CCNC(=O)C1.C12CCC1CC(=O)N2 CC(C)C1=NOC(C)(C(N2CC3CCC2CN3C(C2CN3CCC2CC3)=O)=O)C1 O=S(=O)(c1cccc(=NC2CCN(CC(F)(F)F)C2)[nH]1)N1CCOCC1 N1(C(CC2CC(OCC)C2)=O)CCC2(CCN(C(c3cncs3)=O)CC2)C1 c1(CNC2CCCC(C(=O)NCc3cn[nH]c3)C2)cc(Cl)cnc1F O=C1NC2(C(=O)NC3CC(NC(=O)CC(Cl)Cl)C34CCC4)CC3CC1C2C3 C(=O)(C1(C)CCOc2ccccc21)N(C)CCNC(C1CC2C=CC1O2)=O c1(CC)nn(C)c(CC)c1C(=O)NCC(C)(C)CN(C(=O)CCCC#N)C C(=O)(CCCC(=O)N1CCC(C=O)C1(C)C)NC.N1(C(C)=O)CC(OC)CC1=O CCC(CC(=O)N1CCC(C(=O)NCC(C)(C)CSC)C(C)(C)C1)C(F)F N1(C(C(C)(C)N2CCCC2)=O)CC2CC(NC(c3sccc3N(C)C)=O)CC1C2 c1(SC)ccnc(NC2CCN(C(c3ccco3)=O)CC2)n1 Cc1ccc2c(C(N3CCCC3C(=O)Nc3ccc(I)nc3)=O)c[nH]c2c1 C(=O)(C(CNC(C1CCCO1)=O)CC(C)C)N(C(C(=O)OCC)C)C1CC1 N1(C(C=CC=CCC)=O)CCC(NC(=O)CC2CC3(CCCC3)CO2)C(C)(C)C1 C1(OC)CCn2cc(C(=O)NCC3C(C)CCN3C(=O)CN3CC=CC3)nc2C1 C(CC(C(=O)NC(C1CCN(C(=O)C(C)N(C)C)C1)C)NC(C)=O)SC Cn1nnc2ccc(C(=O)NCC3CN(C(=O)CCC(N)=O)CC(C)(C)C3)cc12 c1(C(N(C(CN(C(C(CC(C)C)O)=O)C)C)C)=O)cc2ccsc2n1C Cc1cc(C(N2CCC(CNC(c3csc(Br)c3Cl)=O)C2)=O)[nH]c1C N1(C(c2c(CC)ncs2)=O)CC2CC1CN(C(=O)C(C)c1ccsc1)C2 CC(CCO)CCN=c1nc(N2CCN3CCOCC3C2)c2cc(Cl)ccc2[nH]1 C(=O)(C(O)C(C)(C)SCCOC)N(CCNC(C(C)(C)NC(=O)OC)=O)C(C)C CC1CCCN(CCCN2CCCC(CNC(C3CCCCO3)=O)C2)C1 Cc1cc(F)c(C(=O)NC2CCN(C(=O)Cc3cccc(F)c3)CC2C)cc1F c1(C(N)=O)cc(-c2ccc(C(=O)NCCCOCc3ccccc3)o2)ccc1Cl C1(CCC)CCC(C(=O)NC2CC(NC(=O)C=CC3CCOC3)C(O)C2)CC1 N1(C(C(CC)(C)CC)=O)CCC2(C1)CN(C(C13COC(CCO1)C3)=O)CC(C)O2 C(=O)(C(CCOC)NC(=O)CC1CC(C2CC2)C1)N(CC(COC)O)C c1(CC)ccc(C(N2CCC(CNC(=O)Cn3cc(CO)nn3)C2)=O)c(OC)c1 C=CCC(CC(F)F)C(=O)NCC(c1cccc(C)c1)NC(=O)C(C)S(C)(=O)=O c1(CN(C)C(=O)NCc2cc(C3CC3)on2)cnn(C(C)C)c1 C(CC(=O)N1CCN(C)C2(CC2)C1)(C(C)(C)C)NC(C(C)=C1CC1)=O N1(C(c2nc(C)c(Br)cc2)=O)C2CCCC1CC(n1ccnc1)C2 c1(NC)ccccc1C(=O)NCCC(O)CNC(=O)C=CCCC(C)C N1(C(CC2ON=C(C)C2)=O)C(C(=O)NC2(CO)CC(O)C2)CCC1C(C)C C#CCCCCCC(=O)NCC(C1CC1)Nc1ccc(OC)c(OC)c1 c1(C(=O)NC2COCC2C(=O)Nc2ncccc2CO)cnc(O)nc1O C1(NC(c2cc(C)sc2)=O)C2CCN(C(=O)CC3(C#N)CC3)C12 c1(C(N2CC(NC(CCC(CC)OC)=O)(CC)C2)=O)ccc2ncccc2c1 C1(NCc2c(OCCOC)ccc(Cl)c2)CCC12CCCCC2 c1(C(N2CC(NC(C34CCCCC3C4Br)=O)C2)=O)sc([N+](=O)[O-])cc1Cl C(N=c1[nH]c(Cl)c(CC)s1)C1(C(=O)OCC(C)(C)CC(=O)NCC)CCC1 c1(C(N2CC(NC(c3cc(C)sc3C)=O)C2)=O)ccnc2ccc(F)nc12 C12(C(=O)OCC)C3C4C1C1C2C3C41NC(=O)N(C1CCCCN1)C C(=O)(C(Cc1cn(-c2ccncc2)nn1)NC(C1CCN1S(C)(=O)=O)=O)OC C1(C(N2CCCC(CCC)(NC(c3csnn3)=O)C2)=O)Cc2cc(F)ccc2O1 c1(OC)cc(C(=O)NC2CCC2NC(C2CC23CCSCC3)=O)cc(F)c1 NS(=O)(=O)c1ccc([N+](=O)[O-])c(NC(=O)C(F)=C2CN(c3ccon3)C2)c1 N#Cc1ccc(Br)c(F)c1C(=O)NCC1CCN(C(c2cc(Br)ccc2O)=O)C1 C1(CCC)(NC(=O)Cn2c(C)csc2=O)CCCN(C(C2(C#N)CC2)=O)C1 CCCCC(C)C(C(=O)NCC(=C)C)N1CCc2cc(C(F)(F)F)ccc21 N1(C(=O)OC(C)(C)C)CCN(CC2CCc3ccccc32)C2(CCCC2)C1=O C1(CCNC(CN(CC)CC)=O)CCCN(C(c2c(C)oc(C)c2C)=O)CC1 c1(OCC=C)ccc(C(=O)NCC(C)N(C(=O)CN2CCC2C)C)cc1 N1(C(N(c2ncc(C#N)cc2Br)c2nc(COC)cs2)=O)CCc2sc(Br)cc2C1.O=C.O Cc1ccc(C(=O)NCC(=O)NCCNC(=O)CC(C)N2CCCC2=O)s1 C12(CNC(=O)C(F)CC3CCC3)CCC(C1)N(C(c1cnn(CCF)c1)=O)C2 N1(C(C=C(C)C)=O)CCC2(CC1)CCN(C(=O)C(C#N)CCc1ccccc1)C2 C1(NC(=O)Cc2cccs2)CC2CC1N(Cc1cc(Br)c[nH]1)C2 N1(C(CC=CCC)=O)CCC(OCC(=O)NCCF)C1 Cc1cc(C)c(C(N2CCC(N(C)C(C3CC(CCO)C3)=O)C2)=O)cc1C CCC(CC)C(F)C(=O)N1CCCC1CN(C)C(c1cc2n(n1)CCCN2)=O N1(CCNC(C(C)N(C)Cc2ncc(-c3ccccc3)o2)=O)CCOCC1=O C1(C(=O)NC(C(C)C)CCO)CN(C(=O)C=CC2CCC2)CC1(F)F C1(C(=O)Nc2nc(C)c(C)s2)C2CCC(C2)C1NC(c1cnnc(O)c1)=O CCCC(C(=O)N(C(C)CN(C(=O)CCc1cc(Cl)no1)C)C)c1ccccc1 c1(SCC(=O)NCCC(C)(C)NC(CCC=C=C)=O)cc(=O)n2ccsc2n1 C1(CC(=O)N(C)CC2CCCC2)CC(F)CN1C(c1ccc[nH]1)=O C(C)(C(=O)NCCC1(O)CN(C(=O)CCCSC)C1)(C1(C)CC1)OC C(=O)(C(O)CC[S+](C)C)NC1CC(NC(C2C(C#C)C2(C)C)=O)C1 N1(C(CC2CC(NC(C)=O)C2)=O)CCN(C)CC1CN(C(=O)C=CSC)CC c1(C(C(=O)N(C2(CCN(C(C3CCC4CC34)=O)C)CC2)CC)(F)F)ccc(Cl)cc1 Cc1cccc(O)c1C(N1CC2CCC2(CC(N2CC(O)(C(N)=O)C2)=O)C1)=O CCCC(C)(C)C(=O)NCC(O)CCNC(C1CC(C(F)(F)F)(OC)C1)=O c1(C(=O)NC(C)(C)CCNC(C2CC23CC3(F)F)=O)nccc2cccnc12 C(=O)(CC(C)C(=O)NC1(CNC(C2CC(C)OC2C)=O)CC1)OCC N1(C(C(C)(C)NC(=O)OC)=O)C2CCC1C(F)C(NC(=O)CC(F)(F)C(F)F)C2 c1(C(N(C(c2cc(C(C)C)on2)C(=O)NC2COC2)CCC)C)ccccc1F N1(C(c2ccccc2)=O)CCC(O)C(C(N2CCCC(n3ccnn3)C2)=O)C1 CS(=O)(=O)c1ccnc(NC2CN(C(c3ccc(I)cc3)=O)CC23CC3)n1 Cn1cc(C(N2CCC(NC(=O)C=CSc3nc[nH]n3)C2)=O)cn1 c1(NC(CC)=O)cc(C#N)ccc1-n1cc(CN2CCCCCC2)nn1 C1(C(=O)NC(CSCC)C(=O)NC(C)C(C)F)OCCC1(C)C C1(C)(CNC(C(CCC)N(C)C)=O)CCCN(C(=O)Cc2cc(C)cs2)C1 CC(C)CCCC(=O)N1CCCCC1C1(C(=O)N(CCCO)CCO)CC1 C1(C(=O)NCC2CC(CNC(C3C(C)(CC)C3)=O)C2)C2CCC1CC2 C1(COC)OCCC1(C)C.C12(C(CO)CN3C4(CC(F)C4)C3=O)CCC(CC1)C2 c1(C(N2CC(C)(C(=O)NC(CCC)c3ccco3)C2)=O)[nH]cc(C)c1C Cc1cc(C=CC(=O)NCC2CCN2C(=O)C(c2cnn(C)c2)C)ccc1F c1(C(=O)NCC2CCN(Cc3n(C)ncc3Br)CC2)cc2ccccc2cn1 NS(=O)(=O)CCCC(=O)N1CC(O)C(O)C1CNC(C1CC2CC2C1)=O c1(C(=O)NC2CCN(C(c3cc(Br)cc(Br)c3)=O)C2)noc2c1CCCCC2 C1(CNC(c2cc(CCC)sc2)=O)(NC(c2c[nH]nc2CC)=O)CCOCC1 c1(C(=O)NC2CC(O)(CNC(C3(CC)CCCC3)=O)C2)ccc(S(N)(=O)=O)nc1 N1(C(CNC(=O)NC)=O)CCC2(CC1)CC2(CO)CNC(c1ncccc1C)=O C1(CC)COC(C)CN1C(=O)CCN(C)C(C1CN(C(N)=O)C1)=O C#CCCCCCCC(=O)NCC1CN(C(=O)C(C)(F)c2ccccc2)C1 c1(C(=O)NCCOC2CN(C(=O)CCOc3ccccn3)C2)cnc(S)nc1 C1(C(CCC)OC)(OCCOCC)CCCN(C(=O)C(N)=O)C1.C1(C)C(=O)N1 C1(C(=O)NCC2(C#N)CCC2)(COC)CN(C(c2ccc(C)o2)=O)C1 CCC(C)(C)CCCC(=O)NC(C)(C)CNC(c1cc([N+](=O)[O-])ccc1OC)=O N1(C(C2(SC)CC2)=O)CCC2(COCC(CNC(C3(NC(C)=O)CCC3)=O)O2)C1 c1(OC)ccc2c(c1)CC(C(=O)NC(C)CN(C)C(c1cccc(O)c1F)=O)O2 Cc1ccc2scc(C(N3CCC(C)C(NC(=O)Cc4cscn4)C3C)=O)c2c1 c1(C(C)N(C)C2CC2)ccc(Cl)c(Cl)c1.C1(C)CCN(C(=O)COCC)C1 Cc1cc(F)cc(C)c1C(=O)NCC#CCNC(C1(C(C)C)CCC1)=O C1(NC(C2C(c3cc(C)sc3)C2)=O)CC2CCC(C1)N2C(=O)C(N1CCSCC1)C C#Cc1ccc(C(=O)NC(C(=O)NCC2CC2(F)F)C(C)C)o1 CC1CCCC=C1C(=O)NCCCCCNC(=O)Cn1ccc([N+](=O)[O-])n1 Cc1ccc(C#N)cc1S(=O)(=O)N1CCC2C(CCN2C(c2cc(C)[nH]n2)=O)C1 C12(NC(c3cnn(C)c3Cl)=O)CC3CC(C1)CC(CNC(C1CCC1)=O)(C3)C2 c1(C(N2CCC(C)(CNC(C(CCC)C(C)C)=O)C2)=O)nnc2ccccc2n1 C1(CNC(C2OCCN(C(C(C#C)(C)C)=O)C2)=O)CCC2(CCC2)O1 C#CC1(O)CC(C(N2CC(NC(c3nccn3CC)=O)C(CO)C2)=O)C1 CCCCC(C)(F)C(=O)NCCOC1CCN(C(c2cncc(F)c2C)=O)C1 C1(NC(c2ccc(COC)[nH]2)=O)CN(C(=O)C=C(Cl)Cl)C2CC12 S(=O)(=O)(c1ccc2[nH]c(=NCC(CO)OC)sc2c1)NC(COC)CO N1(C(c2ccc(OC)o2)=O)CCOC(C(=O)NOC(C2CCCC2)C)CC1 C1(C(N(C)CC2CN(C(=O)CCc3ccon3)CCO2)=O)CCc2ccnn2C1 c1(C(=O)NC2C(NC(CC3(OCC)CCC3)=O)COC2)ccc(CC)c(F)c1 CCC(CCC(=O)N1CCC(C(=O)NCc2ccc(F)cc2O)C1(C)C)OC CCC(C)C(C(=O)NC(c1ncc(C)cn1)C)N(C(=O)C=C(C)C(C)C)C C#CC1(NC(=O)CC2CN(C(=O)C(CC=C)OC)CC23CC3)CCC(C)(C)C1 c1(CC(N2C(C(=O)NC(C)CCc3cn[nH]c3)C=CC2)=O)ccc(O)cn1 C1(NC(=O)C=CCF)CC2CC1N(C(c1csc(-c3cnc[nH]3)n1)=O)C2 c1(CSC)noc(C(C)NC(=O)C(=O)NC2CCN(S(=O)(=O)C(F)F)C2)n1 C1(NC(C(c2ccc(Cl)s2)C)=O)COCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 n1(CCC(=O)NCC2(F)CC(NC(CCC3(C)CC3)=O)C2)cnc([N+](=O)[O-])c1 N1(C(C(N2CCN(c3ccc(Cl)cc3)CC2)=O)=O)CCC(F)C(O)C1 C1(C(CC)C)CCN(C(c2cc(CNC(C3CCC(C)(C)OC3)=O)no2)=O)CC1 Cc1ncc(C(=O)NCc2ccc(C(=O)N(CCCN(C)C)C)nc2)n1C c1(NC(C2(c3ccccc3)C(C)C2)=O)ccc2c(c1)CN(C)C2 CC(CCN=c1[nH]c2c(c(=NC(CN(C)C)CCO)[nH]1)COCC2)c1ccccc1 Cc1ncccc1-n1c(S)nnc1-c1cccnc1.C1(C)CCOC1 c1(C(=O)NCC2(CN(C)C(C34CCC(C3)C4)=O)CC2)coc2c1COC2 c1(C(=O)NCC(C)NC(C(c2cccc(C)c2F)O)=O)cc2n(c1)CCOC2 c1(CC)cc(C(N2CCCC2C(=O)NCC2CC(O)CN2)=O)cc(Cl)n1 n1(CCC(=O)NCC2(OC)CN(C(c3cc(C)c(C)o3)=O)C2)cc[nH]c(=O)c1=O c1(OC)cc(SC)ccc1C(=O)NC1CCN(C(=O)Cc2cccnc2)C(C)C1 N1(C(c2nc(C)oc2)=O)C2CCCC1CN(C(c1nc(C3CC3)ncc1Cl)=O)C2 C(=O)(CCCCCC(C)O)NCCCN(C(C(CC)c1cccnc1)=O)CC c1(NC(C(=O)NCc2n(CCC)ccn2)=O)ncc(C)cc1F C(=O)(CC(C)C(C)(C)C)N1CC(CNC(COCC=C)=O)C(C)CC1 C(=O)(C1=C(C)CCCC1)NCC(CC)NC(=O)CN(CC)CC c1(C(C)C)cc(C(N2CC3CC3(NC(c3cscn3)=O)C2)=O)ccc1F N1CCc2cc(Br)cc(F)c21.Cc1nn2cc(S(=O)(=O)N(C)C)nc2s1 c1(NC(CC2CCC(NC(C=C(C)C)=O)CC2)=O)cc2[nH]ccc2cc1C#N CCCC(C(=O)N1CCCC1C1(O)CN(C(c2ncn(C)c2C)=O)C1)OCC N1(C(C(CCC)O)=O)C(CNC(c2ccc3c(c2)NCC3)=O)CC2COCC12 Cc1cnc(C(N2CCC2C(=O)N(C)CCn2cc(C)cn2)=O)c(F)c1 N1(CC2CCC(C(=O)OCC)O2)CCCC2(COc3ccccc32)C1 N1(C(C=C(C)C)=O)Cc2occ(C(=O)Nc3cnn(CCF)c3)c2C1 C(=O)(C(C)(C)C(N)=O)NC(C(=O)NCCC(C)F)C C=CCC(CNC(=O)Cc1ccccc1)NC(=O)C(C)=CC=CC(C)(C)C O=C(C1CCCc2nc[nH]c21)NC1CCN(C(=O)CCCn2cccc2)C12CC2 N1(C(C2C(C)(CC)C2)=O)CCCCC12CN(C(=O)Cc1sc(O)nc1O)C2 c1(NC(C2N(C(C3(C)CC3)=O)CC(F)C2)=O)ccccc1N1CCCCC1 c1(C(N(CCCNC(C2CC(=O)N(OC)C2)=O)CC)=O)csc2ncnc(O)c12 c1(C(=O)NC2(C)CCN(C(c3c(C)cnn3C)=O)CC2)cnc2c(c1)NCC2 C1(c2nnnn2C2COC2)(NC(CC)CC2CCCC2)CN(CC)CC1C C(C(=O)NCC12CCCC1OCC2)(C(C)(C)C)NC(CSCCC(C)C)=O C1(O)(N(C(C(C)NC(C)=O)=O)C)CCN(C(C2(CC(C)C)CCCC2)=O)CC1 C1(CNC(=O)OC(C)(C)C)CC2CCC(C1)N2C(N)=O.C1(CF)CCC(=O)N1 CC(C)CCCC(C)C(=O)NC(C1(O)CCN(C(C2CCCC2(C)C)=O)CC1)C Cc1nc2ccc(C(N3CCC3CNC(c3cncc(Cl)c3Cl)=O)=O)cc2nc1C N1(C(C)=O)CCOCC1NC(C(=O)NC(Cc1ccccc1)CCNC(N)=O)C C1(C(=O)NC(CCSC)C(=O)NCc2cccc(F)c2)CC2CC(=O)C1C2 S(=O)(=O)(c1cccc(=NC(C)CCCO)[nH]1)NCC1(SC)CCC1 C1(C(=O)NCC(C)(C)NC(=O)CSc2nc[nH]n2)CCCCC1C1CC1 C(=O)(CCCS(N)(=O)=O)N1CCC(N(CCC)C(c2cc(F)cc(F)c2)=O)CC1 C12(C(N(C(C(C)C)C)C)=O)CC(CO)(CN1C(=O)CC1CCN(C)C1)C2 N1(c2snc(CCC)n2)CC2C3CCC(C2C1)N(C(=O)C#CC1CCCCO1)C3 N1(C(Cc2ccc(C)s2)=O)CCOC(CC(=O)NCc2cncn2C2CC2)C1 N1(C(c2c(CC)nnc(C)c2)=O)CC2CCC1C(CO)C2 C12(NC(C(C)C3CCC3)=O)CC(C1)N(C(=O)COCc1cccnc1)C2 Cc1cc(F)cc(C)c1C(N1CC(C(C)NC(c2nnn3ccccc23)=O)C1)=O C(CC1=CCN(C(=O)CC2CCC2OC)CC1)NC(CC1(OC)CCOCC1)=O N1(C(CC2CC(=C)C2)=O)CC(C2CN(C(c3cncc(F)c3)=O)C2)C1 C1(F)(C(=O)NCC(C)N(C)C)CCN(C(C2CCC(C)(C)C2)=O)CC1 C(=O)(C(C)CCOC)NC1C(C(=O)NCC2(C#C)CCC2)CCC1 C1(C(N2CC(NC(=O)Cc3cncn3C3CC3)(CO)C2)=O)OCC2CCCC12 C(=O)(C(=O)CC(C)C)NC(C1CCCC1)CNC(c1cc(C)no1)=O N1(C(Cc2c(C)ncs2)=O)C(CNC(C23CCC(CC2O)C3)=O)CC2CCCC12 C(c1ccc(NS(C)(=O)=O)cc1)=CC(N1CC(NC(c2nc(C)sc2)=O)C1)=O N1(C(C(CCC)F)=O)CCC(C)C(CC(=O)Nc2cn(C)nc2SC)C1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCC1C(NC(c1c[nH]ccc1=N)=O)C2 c1(NC(c2ccncc2Br)c2n(CCSC)nnn2)cc(C(F)F)cc(F)c1 n1(CC)cnc(C(=O)N(C(C(=O)NCC2(CO)CC2(C)C)C2CC2)C)n1 C#CCC(C)(C(=O)NC(C)C(O)C(F)F)NC(c1cnsc1)=O C=CC(CCC)CC(=O)NCC1(OC)CN(C(c2c(C)ccc(Cl)c2N)=O)C1 Cc1cc(C(=O)NC2CC(CNC(=O)C(C)C3CC3)C2)c(Br)cc1F C1(NC(C2CCCN2)=O)CN(C(c2ccc(Br)s2)=O)CC12CCCCC2 Cc1cccc2[nH]c(C(N3CCN(C(c4ccc(F)cc4N)=O)C4CC34)=O)cc12 CC(O)(CNC(=O)Cc1csc(-c2ccco2)n1)CNC(=O)CC#N C1(C(=O)NC2CCN(C(C(CCC#C)O)=O)CC2F)CCC2CC1C2(C)C c1(C(=O)NCC2C(CNC(C3CNC(=O)N3)=O)C2)cnc2n1CCOC2 C1(C(=O)NCC2(C)CCN(C(=O)Cc3ccon3)C2)CCc2cnnn2C1 c1(C(=O)NC2CC(NC(c3ccc4c(n3)CCC4)=O)C2)ccc(F)c2occc12 c1(-c2sc(NC(N(CC(C)O)CC)=O)c(C)n2)nc2ccccc2s1 c1(C(CCC(=O)NC(CCNC(C(C(C)C)O)=O)C)=O)ccc2c(c1)CCC2 C1(NC(=O)C2CC2)CN(C(c2occ3c2CCCC3)=O)CC(F)(F)C1 N1(C(Cc2ccc(OC)cc2F)=O)CC2CN(C(=O)C=Cc3cscn3)CCC12 CC1CCOCC1C(N1CCCC1C=CC(=O)NC1COCCOC1)=O Cc1cccc2c1CCOC2C(=O)NCCCNC(=O)CCCF C1(C(=O)NCC(C)(C2CC2)NC(c2cc(OC)no2)=O)CCN(C)C(=O)C1 Cc1ccc(COCC(=O)NCC(C)NC(=O)CNC(=O)NC2CC2)cc1F.OC c1(CCCOC)nc(C(n2cncn2)C)n(-c2cccc(F)c2)n1 c1(C(=O)Nc2cc(OC(C)C)n[nH]2)ccc2ncc(-c3cc(O)c(F)cc3F)n2c1 C1(CNC(CC(CC)OC)=O)COCC(=O)N1C.C12(CCN(C(C)=O)C1)C(=O)O2 c1(C(=O)NCCn2cc(CCC(=O)O)nn2)cc(F)c(F)cc1Cl N1(C(Cn2c(C)cc(C)n2)=O)CC(C)CCC1CNC(C1(CO)CCOCC1)=O c1(C(N(C(C)CCNC(c2ccc(CO)s2)=O)C)=O)cc(N)cc(O)c1 N1(C(c2c(C)cns2)=O)CC(C)(C)OCC1CNC(=O)COC1(C)CCOCC1 N1(C(COC(CNC(CNC(C)=O)=O)(C)C)=O)CCOCC1CCO c1(C(C)=O)cc(C(=O)NC2(CCNC(=O)C(F)C3CCCC3)CCCC2)oc1C c1(CNC2(c3nnnn3CCCF)C(C)SCCC2)nc2cc(Br)ccc2s1 CN=c1nc(N2CC3CCOC3C2)[nH]c(=NCCS(=O)C(C)(C)C)[nH]1 N1(C(C(COC)NC(=O)C(C)OCC2CC2)=O)CCC(C2(OC)CC2)C1 C(CCN=c1nc(N2CCC(CN(C)C)CC2)c2sccc2[nH]1)c1cc(C)no1 CC1OC(C)CC1CC(=O)NCCOCCN(C)C(C1(CO)CC(F)(F)C1)=O N(C1CCCc2occc21)C(CCN(C(c1c(NC)cnnc1)=O)C)=O CCC(CCCC(=O)NC1CCN(C)CC1(C)C)NC(C12CC(CO)(C1)C2)=O C(CNC(c1c(C)ncn1C)=O)(C(C)(C)C)NC(c1cc(CSCC)on1)=O c1(C(=O)NC2(C)CCN(C(CC(C=C)C)=O)C2)cc(OC(F)F)cc(Br)c1 c1(OC)cccc(C(CF)N(C)C)c1.C1(C2C(=O)O2)CCCCO1 C(=O)(C1=CS(=O)CCC1)N1CC(=CCNC(=O)OC(C)(C)C)C1 N1(C(NC(=N)N)=O)CCOC2(C1)CN(C(c1ccc(CC3CCC3)cc1)=O)C2 c1(C(N2CC(N(C(C(CCC)c3ccccc3)=O)C)C2)=O)cc(C)c(F)cc1N C(CC(=O)NC)(C(C)N1CCC2CC12C(=O)OC)NC(C(CC)C#N)=O C1(CNC(C#CC(=O)N(C)C)=O)CCN(C(c2ccc(O)c(F)c2)=O)CC1O C(=O)(CC(C)(C)C)NC(C)C(N1CCC(O)(C(C)NC(=O)CO)C1)=O CCCCC(C(=O)NCCC(O)C(C)C)NC(=O)CN1CCCCC1C c1(C(Cn2c(N3CCC(c4cncc(C)c4)CC3)nnn2)C)ccc(Cl)cc1F N1(C(CC(=O)OCC)=O)CC2CCCN(C(C3CC(F)(F)C3(F)F)=O)C2C1 c1(CNC(C2(C)CC(C)OCC2)=O)nc2c(s1)CN(C(=O)C(C)(F)F)CC2 n1(CC#C)c(C(N2CCN(C(=O)CSC)CC2C2CCC2)=O)cc2ccccc12 CC(C)(F)CCC(=O)NC12CCOC(CNC(C3CS(=O)(=O)CCO3)=O)(C1)C2 CC(C)(C(=O)NCCC1CCC(CC)C1)C1CCCC1.C1(O)(C(=O)N)COC1 CC1=C(C(=O)Nc2nccc(N3CCOCC3)n2)C(C)(C)CCC1 Cc1nn(C)c2ccc(C(=O)NC3CC(NC(C4CCC(F)(F)C4)=O)C3)cc12 C1(C(N(C(CC)CSC)C)=O)C(C)OCCN1C(=O)C(C)NC(C)=O N1(C(c2ccc(CN(C)C)nc2)=O)CC(NC(C2COCCO2)=O)CC12CCC2 C1(C(F)(F)F)(C(=O)NCC(N(C(C(C)OC)=O)C)C2CC2)CCCCC1 C1(CNC(C(c2cnccn2)C)=O)CCC(NC(=O)C(c2ccnn2C)O)CC1 C1(NC(C(CC)O)=O)(CO)CCCN(C(c2nc(C)n(C)c2C)=O)C1 c1(NC2CC(C)CN(C(=O)NC3CC3)C2)c2c(nn1-c1ccccc1)CCCC2 n1(C(C(=O)NC(C(C)C)CNC(=O)C2=CCCC2)(C)C)cc([N+](=O)[O-])cn1 C1(NC(c2c(C)cc(C(F)F)o2)=O)CC12CCOC(C)C2.C12(O)CCN(CC1)C2 N1(C(C(CC=C)CC)=O)CCCC2(C1)CN(C(c1ccc(C)c(C)c1Cl)=O)C2 C(=O)(CCCCC(C)=O)NCc1c(C(N(CC)Cc2c(C)cnn2C)=O)occ1 C1(NC(CSCCC)=O)CCCC12CN(C(c1cc(C(=O)OC)cc(O)c1)=O)C2 C(CN=c1nc2ncn(C)c2c(NC)[nH]1)NC(CN(CC)Cc1ccsc1)=O C[Si]1(C)CCCCN(C(=O)C(=O)NCc2cccnc2Cl)C1 Cc1ccc(C(=O)NCC2CC(NC(C3(C)C=CCC3)=O)C2)cc1F N1(C(N)=O)CCC(C(N2CCCC(N(CCO)C(c3nccnc3N)=O)C2)=O)CC1 c1(CC)cc(C(=O)NC2CC(NC(C3CC34CCCC4)=O)C2)nn1C c1(C(=O)NC(CN(C(CCC)=O)CC)C)ccc(Oc2ccccc2)cn1 C(=O)(CC(CSC1CC1)NC(=O)CSC)N(CCCCO)CC#C C12(C(=O)NCCN(C(c3cn(C)[nH]c3=N)=O)C3CC3)CCN(CC1)CC2 C(C)(CCC(=O)N1CCCCC1CNC(C1(CCF)CC1)=O)SC c1(NC(=O)CCC2CCOC2)cc(C(=O)NCc2cnsc2)no1 N1(C(c2c(C)cccc2)=O)CCCN(C(c2coc(Br)c2)=O)C(CO)C1 CCCC(C(=O)OC)C(=O)N1CCC1CC(N1CCC(OC2CC2)C1)=O C12(C(N3CC(N(C(C4C(C)CCO4)=O)C)C3)=O)CCC(CO1)C2 C1(C(=O)NCC2CN(C(CCOC)=O)C2)CN(OC(=O)NC(C)(C)C)CCO1 C1(CC(C)C)CCN(C(=O)CNC(=O)CNC(c2ccc[nH]2)=O)C1 Cc1c(C(=O)NCC2CC2NC(=O)CSc2nnnn2C)ccn1C(C)C CC(C)C(CCNC(C1CC1Cl)=O)NC(C12CC3CC1C2C3)=O C1(NC(CCC=C(C)C)=O)CCC2CN(C(=O)Cc3ccc(Cl)s3)CC2C1 C1(C(=O)NC2C(CC(=O)O)COCC2)(C(=O)O)CCS(=O)(=O)CC1 C1(OC)CN(C)CCC1NC(c1sccc1Nc1nccc(C)n1)=O Cn1cc(C(N2C3CCC2C(CNC(C2COC(=O)N2)=O)C3)=O)ncc1=O CC(C)C(C)C(C)CC(=O)NCC1CC1CNC(=O)C(C)(C)c1ccnn1C c1(C(=O)OC)cc2n(n1)CCCC2NC(=O)OCCCOC(=O)CO c1(CNC(=O)OC(C)(C)C)cc(F)cc(Br)c1.C12CC(C1)NC(=O)N2C1CC1 C1(C)(C(=O)NCc2c(C(=O)NCC)c[nH]n2)COC(=O)N1 N1(C(C2(O)CCC2)=O)CCCC(F)(C(N2C3CSCC2C3)=O)C1 C(=O)(CCC(=O)NN(C)C)N1C(CCC(=O)NC(C2CCCC2)CC)CCCC1 CN1CC(C)(C)CC1C(N1CCC(F)CC1C(=O)NC1(n2cccn2)CC1)=O Cc1nc(=NCC2CCCC(NC(C3(C(=O)N(C)C)CC3)=O)C2)[nH]cc1[N+](=O)[O-] CC1=C(C(=O)N2CC(N(C)C(c3ccco3)=O)C2)CCCC1 c1(C(N(C2CCN(C(=O)CCCC(F)F)C2)CCO)=O)nccc2ccncc12 C12(NC(c3ncc(OC)cn3)=O)CCC(C1)N(C(C1(n3cccn3)CC1)=O)C2 c1(NC(C2C(NCc3c(F)ccc(C#N)c3)CCC2)=O)ccc2oc(O)nc2c1 N1(C(=O)O)CCSC2COCCC12.Cc1cccc(OC(C)(C)C)c1 c1(C(=O)NC2(CC=C)CN(C(c3snc(C)c3N)=O)C2)cc(F)c(F)c(Cl)c1F N1(C(c2c(CCC)nns2)=O)CCCN(C(=O)CNS(N)(=O)=O)C(CO)C1 N1(C(c2cn(CCC)nn2)=O)C(C(N2CCNC(=O)C2C)=O)CCC12CC2 C12(C(N3CC(CN(C(C(CCC)NC(C)=O)=O)C)C3)=O)COCC(C1)OC2 N1(CC(=O)NCC2N(C(C(CCC#C)O)=O)CCC2)C(=O)c2cccnc2C1=O C1(NC(C2C(CCC)C2)=O)COC2(CCN(C(c3cccs3)=O)CC2)C1 c1(CC)ocnc1C(=O)NCC1(F)CC(NC(=O)C(C)OCCC(C)C)C1 c1(-c2n(CCCOC)nc(CCC(C)(C)C)n2)ncc(Cl)cc1Cl N1(C(c2n(C)c(=O)ccc2)=O)CCC=C(C(=O)Nc2cc(F)c(F)c(F)c2)C1 N1(C(C2CCC(=O)C2)=O)CCCC(C(N2CCC(OC3CC3)CC2)=O)C1 CCC(CCCC(=O)NC1CCC(CCO)CC1)NC(=O)C(C)O C(=O)(C(C#N)(CC)CC)N1CC2CNC2C1.c1(-c2nc(CC)on2)cc(Cl)cnc1Br C1(NC(=O)CCn2ccnn2)CN(C(c2ccon2)=O)CCC1C(F)(F)F C1(C(=O)NCC(C=C)O)(SC)CN(C(=O)CN2CC=CC2)C1 C1(=O)C(CC(N)=O)N1.C(=O)(C(C)C=C=C)N(C(CC#C)C)C c1(C(=O)NCCC(C)NC(c2nnc(O)nc2O)=O)ccc(CO)c(F)c1 C1(CN(C)C(c2cocn2)=O)CCCC(NC(c2ccc(C(F)(F)F)cn2)=O)C1 CCC(CC)C(=O)NC1CCCCC1CNC(c1ccccc1Br)=O C12(CC)CN(C(C3CC3SC)=O)C(COC)(C1)C2.c1(C(=O)NC)cncnc1O.SC CC(C)C(CO)C(=O)NC(C1CCCCC1)CNC(c1cnc(Cl)c(Cl)c1)=O CCCC(O)CC(=O)NC(CO)C(C)NC(=O)CCCc1cncs1 C1(CC(=O)NC(CNC(C2CC(=O)NC2=O)=O)C2CC2)C2CC3CC(C2)CC1C3 C(=O)(C1CCCc2n[nH]cc21)NCCN(C(c1cc(C)nc(C)c1O)=O)C c1(C(C)O)cccc(F)c1.n12cc(nn1)CN(CCN(C)C)C(=O)C2 C=C1CCC(C(N2CC(OC)CC2CNC(=O)C(CCC)NC(N)=O)=O)CC1 c1(C(N2CCC(CN(C(C=CC(C)=O)=O)C)C2)=O)ccc2nc(O)n(C)c2c1 c1(CC)ccc(NC(=O)CCC(C)NC(C2CCN(OC)CC2)=O)cc1C c1(C(=O)N)cn(CCO)nn1.CC(CN(C(=O)C=CCN(C)C)C)NC C=CC1CCN1C(c1cc(CNC(C2(CO)CCOC2)=O)[nH]n1)=O C1(C(N2CCCC(NC(CCCC#CC)=O)(CC)C2)=O)CCC2(CC1)CC2(F)F C1(C(=O)NCC2C(C(N3CC(CC(C)C)OCC3)=O)CC2)CCCCC1(C)C C1(C2CCN(C(=O)CCn3cncn3)C2)(NC(CCC(=C)C)=O)CC1 C=CC(C)(C)CC(=O)NC(C)(C)C=CC(=O)NC1CCN(C)CC1C N1(C(c2c(N)non2)=O)CCC2CCC(C1)N2C(=O)C(C1CCCCCCN1)F C1(CNC(=O)NC(c2cocn2)CC)CCc2n[nH]c(C)c2C1 N1(C(C(C)OCCOCC)=O)CC(C)(C(N2CCC(C3CC3)CC2)=O)CC1(C)C Cc1ccccc1C=NOCc1sc(C2CC2(F)F)nc1C C(=O)(CCCCC(F)(F)F)N1C(C(C)(C)NC(C2CCC(C)(C)OC2)=O)CCC1 Cc1cccc2c1CC(C(=O)NC1(CNC(c3cc(C)n(C)n3)=O)CCOC1)O2 C(=O)(C(F)(CNC(C1CC(=O)NC1(C)C)=O)C(C)C)NC(C(=O)NCC)CC c1(CC)ccc(C=CC(=O)NC2CN(C(=O)Cn3cccc3)C3CC23)o1 C1(N(C(c2nc(C(C)C)oc2)=O)C)CC2CC1N(C(=O)C=Cc1cn(C)nn1)C2 C1(N(C(CCN(C(C)=O)C)=O)C)CCN(C(=O)C(C)OC2CCCC2)C1 N1(C(C2N(C(c3n(C(C)C)ccn3)=O)C(C)C2)=O)CCCc2occc2C1 C1(CCC(=O)OCC)CCN(C(c2sc(C3CNC3)nc2C)=O)CC1 N1(C(CCC2CC(OC)C2)=O)CC(NC(c2conc2C)=O)C2CCCC2C1 N1(C(c2cc(Cl)c(Br)cn2)=O)CC2CC1CCN2C(=O)CCF C(CC(=O)NCC1(C)CCOCC1)(C(F)(F)F)NC(Cc1c(C)cnn1C)=O c1(NC(C2N(C(c3cn(C)nc3)=O)CCCC2)=O)cc(F)c(Cl)cc1Cl N1(C(c2cc(CNC(C(c3ccccc3)C)=O)[nH]n2)=O)C2CCCC1COC2 c1(C(N2CC(NC(CCCOCC)=O)C(C)(C)C2)=O)c[nH]c2cccc(C#N)c12 c1(N2CCN(CC(Cl)(Cl)Cl)CC2)nccc(=NCc2noc3c2CCCC3)[nH]1 Cc1cc(O)c(Cl)cc1C(=O)NC12CCN(C(c3c(Cl)cccc3Cl)=O)CC1C2 C1(C(=O)OC)CCC(C2CCCCC2)CN1C(C1CC1c1ccco1)=O C1(CC(=O)NCC(COCC)C)CN(C(=O)Cc2c(C)cnn2C)CCC1C N1(C(CCOCC#C)=O)CC2(CCCCC2NC(C2CC3CC3C2)=O)C1 N1(C(c2c(Br)ccc(C)c2)=O)CCC2(CCN(C(c3cnc(O)s3)=O)C2)C1 N1(C(C2CC(OC)C2)=O)CC(C2CN(C(C3COCC3(C)C)=O)C2)C1 C#Cc1ccc(CCCC(=O)Nc2cnn(-c3nccs3)c2)cc1 C#CC1CCCCN1C(c1ccc(CNC(=O)C(O)C(C)C)nc1)=O Clc1cc(CCCn2cncn2)on1 C(=O)(C(O)CCC(C)C)N1CC(C)CC(NC(Cc2nc(COC)sc2)=O)C1 C1(NC(c2c(C)nco2)=O)CCCC12CCN(C(=O)C=C1CCSCC1)C2 C(=O)(CCS(=O)(=O)NC)N1CC(CCC)C(NC(=O)C(C)CN(C)C)C1 c1(C(=O)NC2CC(NCc3nc(C)on3)C2)cc2cccnc2cc1F n1(CC)nc(C(=O)NCCC(C)NC(=O)C(C)CN2CCCCC2)ccc1=O CCCC(C(=O)N(C)CC1CCN(C(=O)C(C)(O)C(C)C)CC1)S(N)(=O)=O C(CCN=c1[nH]c(=NCCC(OC)OC)[nH]c2c1CSC2)C1C(=C)C1 Cc1ccc(C(=O)NCc2cc(F)ccc2Br)c(-n2cc(C(C)(C)C(=O)O)nn2)c1 c1(CNC(c2n(CC)nnn2)c2nccn2C)cc(C(=O)OC)c(C)o1 c1(NC(=O)NC(C)C(C2CCOCC2)C)ccc(C(=O)NC2CC2)cc1 CN1CCN(C(C2CN(C(c3cccc(C#N)c3F)=O)C2)=O)CC1(C)C C(C1CCc2ccccc21)OC(c1cccc(-c2cccnc2)c1)=O Cc1cccc(CCC(=O)NCC2CCN2C(C2CC(=O)N2)=O)c1Cl c1(CC)nnc2n1CCCC2C(=O)NCC1CC1NC(c1ccc(OC)s1)=O C1(CNC(C(CC)O)=O)CN(C(=O)CCn2ccnn2)CC12CC2 N1(C(CC(C)(C)SC)=O)CCC2(CC(NC(=O)C(C)(C)c3cc[nH]n3)CO2)C1 C=CC1(C(=O)NC2CN(Cc3cc(N)c(F)cc3C)CCC2CO)CCCCC1 C1(NC(C(C#C)(C)C)=O)CC2CN(C(c3ccc4cncn4c3)=O)CC2C1 N1(C(C2CCC(OC)CC2)=O)CCC(O)C(C(=O)Nc2cc(Cl)cnc2Br)C1 CN1C2(CCN(CC(F)(F)C(F)F)CC2)C(NC(=O)COC(F)F)CS1(=O)=O N1(C(C2OCCN(C)C2=O)=O)CCN(C(=O)CCCC(F)(F)F)C2CCC12 C(C(C)N)(C(C)C)NC(CC(=C)C)=O.CCCCCC=CC(C(=O)C(F)OC)=O CCC(C)CCC(=O)N1CCN(C(C2COCCOC2)=O)C(C(C)C)C1 N#Cc1ccc(C(=O)NC2C3CN(C(c4coc(Cl)n4)=O)CC23)c(O)n1 Cc1cc(NC2CC(C(=O)Nc3cc(F)ncc3Br)C2)n2nc(C)cc2n1 C(C(C)C(=O)NCC1CC(NC(=O)CCOCc2ccccc2)C1)OCC C1(CCNC(=O)CN2CC=CC2)COCCN1C(c1cccc(C(N)=O)n1)=O N1(C(C2N(C)C(=O)NC2)=O)CCC(C2CCN(C(=O)C(C)(C)CCC#N)CC2)C1 c1(C(=O)NC2(C3CN(C(Cc4ncc(C)s4)=O)C3)CC2)noc2c(F)cccc12 C1(NC(Cc2ccc(C)cc2Cl)=O)CN(C(=O)CN(C)C)C2(CCC2)C1 c1(C(=O)NCC2(CNC(c3nnn(CC)c3C)=O)CC2)ccc(Br)cc1N c1(C(N(CC(C)O)CCNC(CCOC)=O)=O)ccc2n[nH]c(C)c2c1 C=CCC(F)(F)C(=O)N1CCSCC1c1cccc(OC(F)(F)F)c1 CCCCCS(=O)(=O)CC(=O)Nc1cccc(N(C)C(c2cc(C)n(C)n2)=O)c1 c1(SC)ccc(Cl)c(C(=O)NC2CC(CNC(C3CCCN3C=O)=O)C(O)C2)c1 C1(CC(=O)NCC2(C)CCC2)C2CCCC2N1C(C1(C(N)=O)CCC1)=O Cc1onc(Cl)c1C(=O)NC(C)CCCNC(=O)CCCOc1ccc(F)cc1 C(CCC(=O)NC(C1CC=CCC1)CO)N(C)C.C1C(=O)NCCNC1=O C1(CC(=O)NCC(C(C)C)NC(c2cnc(N)c(Cl)c2)=O)CCCCC1(F)F C12(C(N(CCNC(=O)C(C)(CC)CC)CC)=O)CCOC1CCOC2 C=CC1(C(=O)NCC=C2CCN(C(C3CC(=O)N(C)C3)=O)CC2)CCOCC1 C1(CN2CC(CNC(C(CC)SC)=O)C(O)C2)CCCN2CCCC12 C=C(CNC(C1CCC(C)S1)=O)CCNC(c1cn(CC(N)=O)nn1)=O c1(NC(C2C(CC)C2)=O)ccc(C(F)(F)F)c(C)c1.C12CC1N2.C1(=O)CN1 c1(NC(c2c(C)nn(C)c2)=O)ccc(NC(c2ccc(Cl)cc2F)=O)cc1F c1(C(=O)OC)cc2sc(OC(C)C)nc2s1.c12ncn(n1)CC(=O)OC2 C1(C(C)C)C(C(=O)Nc2cnn(C(C)C)c2)CCN1C(C1CCCC2CC12)=O C(=O)(CC1OCc2cc(Cl)ccc21)N1CC2C(NC(=O)CN3CCCCC3)(C2)C1 c1(C(N2CCCCC(N(C(CC(=O)N(C)C)=O)C)C2)=O)c(Cl)cc(Cl)nc1N C(N=c1[nH]c2ccc(Cl)cc2s1)C1CCCC(NC(C2CC(C)OC2)=O)C1 c1(C(=O)OCCOC)ccc(CN(C(C2N(S(CCC)(=O)=O)CCC2)=O)C)cc1 C1(CC(=O)N(CCC#C)C)C2CCCC2N1C(C1CC(COC)C1)=O N1(C(CC(CC)CC)=O)CCC2CC(NC(=O)CCCC(F)(F)F)CCC2C1 C(CC1=CCN(C(=O)C(C)=CC(C)(C)C)CC1)NC(CC=C)=O c1(OC2C(OC)COC2)nc(=NCCC(CO)CC(C)C)[nH]c2ncn(C)c12 Cc1cccc(C)c1C(=O)NCC(F)CNC(c1cc(Br)cn1C(C)C)=O c1(NCC)ccc(C(N2CCC(C)(CNC(=O)CCCOC)C2)=O)cc1[N+](=O)[O-] C1(CNC(C(C)CO)=O)CCCC2CN(C(=O)CC3(N(C)C)CCCC3)CC12 CCCC(C(O)C(=O)NCC(=O)NCC1CC1)NC(c1ccnc(OC)n1)=O C12(CCNC(=O)CCCF)CCC1CN(C(c1ccc(Br)cc1O)=O)C2 C1(C(=O)NC2(C)CC(NC(C3(COC)CC3)=O)C2)Cc2cc(C)ccc2S1(=O)=O c1(CCC(=O)N(C)Cc2c(F)cc(OC)c(Br)c2)nnc2ccc(N(C)C)nn12 c1(C(N(C2CN(C(c3cncc(C)n3)=O)C2)C)=O)cc(F)cc(N)c1N C1(NC(=O)NCc2cc(C(=O)OC)cc(F)c2)CCC2=NN=NN(C2)C1 C1(C(=O)NCCNC(CCCC(C)C)=O)CCC2(CN(C(=O)OC(C)(C)C)C2)O1 c1(NC(N2CCN(c3ccncc3)CC2)=O)ccc(O)cc1 C1(c2nnnn2C2CC2)(Nc2cncc(NC(C)=O)c2)CCN(C)C(C)C1 N1(C(c2c(CCC)n[nH]c2)=O)CCCCC(CNC(c2cc3n(n2)CCO3)=O)C1 CCC1C(=O)Nc2ccc(C(=O)NCCCOCCNC(C3CC3C)=O)cc21 CS(=O)(=O)C1(C(N2CCC23CN(C(c2ccnn2CC(F)F)=O)C3)=O)CCCC1 c1(C(N2CC=CC(NC(C3OCCN(CC)C3)=O)C2)=O)cc2ccc(C)cc2[nH]1 N1(C(C=COCC)=O)CCC(CNC(c2cn(C)c(=O)nc2O)=O)C12CCC2 C1(NC(C2CC=CC(n3cc(CCNC=O)nn3)C2)=O)CC1C1CCCCC1 CCCCCCCC(F)C(=O)NC(C1CN(C(=O)C=NOC)C1)C Cc1ccc(O)c(C(N2CCC(NC(C3(C)CC=CC3)=O)CC2C2CC2)=O)c1 Cc1cc(C(=O)NC(C)CN(C(=O)COCc2cc(C)no2)C)nc(O)n1 c1(OC)ccc(C(=O)N(CC(C)(C)CNC(=O)C(=Cc2cnn(C)c2)C)C)nc1 C123CC(CO1)N(C2)C(=O)CCCCCONC3=O.C(=O)(CCN1CCCC1)OC c1(NC2CC(CNC(c3c(C)nc(CCC)o3)=O)C2)cc2c(cn1)C(=O)CCC2 c1(CN2CC(C(N3CCC(NC(C)=O)C3)=O)C(O)CC2)ccccc1[N+](=O)[O-] C1(C(N2CCOCC2CC2CC2)=O)CSCCN1C(=O)C=Cc1cocn1 C1(CC(=O)N(CCC(=O)N(CC(C)C#N)CC)CC)COCC(C)O1 C(=O)(CC(F)(F)Br)N(C)CC1N(C(c2cc(C)ns2)=O)CCC1 c1(CNC(C2N(CC)CCOC2)=O)ccc(CNC(C2CC2F)=O)c(F)c1 CC1CN(C(C2CNC(=O)CN2C(C2CCC3(CCC3)C2)=O)=O)CC(C)(C)O1 C1(NC(CN(C(C(CC)C)=O)C)=O)C2CN(C(=O)C=CCOc3ccccc3)CC12 C(=O)(C(C)C(O)CC(C)C)N1CCC2(CC1)CC2.C1(NC(COC)=O)CCSC1 CC(C)CC(C)CC(=O)N1CC2CC2C1C(=O)NC1C=CC(CO)C1 c1(NC(C2CCC3(CN(c4ncc5cn[nH]c5n4)C3)O2)=O)ccc2sccc2c1 N1(C(C#CCNC(Cn2c(C)nnn2)=O)=O)CC(C#N)(CCF)C1 C(=O)(CC1=CCOCC1)N(CC(C)O)CCNC(C12CCCC1(C(N)=O)C2)=O C(CCN=c1nc2scnc2c(N2CC(c3ccon3)C2)[nH]1)n1c(O)nnn1 N1(C(C(C(C)NC(c2c(C)non2)=O)C)=O)CC2OC(=O)N(C)C2C1 N1(C(c2c(CC)noc2)=O)CC2(CC(CNC(=O)COC3CC=CC3)C2)C1 c1(C(=O)NCC(COC(C)CO)O)ccc(F)c(C(F)(F)F)c1F Cn1ncc(C(F)F)c1C(=O)NC1CCCCC1NC(=O)C=Cc1ccncn1 C1(NC(C(n2cc(C(c3ccccc3)O)nn2)C)=O)CCOC(c2nccn2C)C1 CC1(C)OC(C)(C)C1C(N1CC(CO)(NC(=O)CC2CCCCC2(C)C)C1)=O C(=O)(C1=NOC2(CCC2)C1)N1C(C)C(NC(=O)C(=O)NCC(F)F)CC1 C1(c2cn(CC3CCC(C(=O)Nc4cnc(C5CC5)s4)C3)nn2)CCCCCC1 CCCC(C)(O)CC(=O)NCCOCCOCCOCCCNC(=O)CN1CCCC1 C(=O)(C(C)(C)CCCF)N1C(C(=O)NC(C)C(O)C(F)F)CCCC1 N1(C(c2cn(CC=C)nc2)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)CC1CF C(=O)(C(C(C)(C)C)NC(=O)C(=O)C(C)(C)C)NCCC(=O)NCC N1(C(CC2(CN)C(C)(C)C2)=O)CC2(C1)CN(C(C1C3CC4C(C3=O)C14)=O)C2.C(O)N C(N=c1[nH]cnc(Cl)c1C(=O)OC)C1OCC(CNC(C=COCC)=O)C1 c1(C(N(C2CCCN(C(=O)C(C)CO)C2)CC)=O)cc(C(F)(F)F)cc(F)c1 N1(Cc2onc(CC(=O)NC)n2)CCC2C(CCCN2C(C2CN(C)C2)=O)C1 N1(Cc2cc3nc(C)sc3cc2)C2CCCC1CC(N=c1c(Cl)c[nH]cc1[N+](=O)[O-])C2 C(=O)(CC(C)C(=O)OC)N(C1CCN(c2nnc(CCOC)s2)CC1)C(C)C c1(C(=O)NC2CN(C(c3n[nH]c(C)c3Br)=O)CC2(C)C)ccc2nn[nH]c2c1O N1(C(C2CSCCN2C(=O)C=CC2CCCC2)=O)CC(CO)C2(COC2)C1 c1(C(N2C(C3(NC(C4C(C5C(C)C5)C4)=O)CC3)CCC2)=O)cc2n(n1)CCCO2 N1(C(c2ncc(OCC)nc2)=O)CCC(F)C(NC(=O)Cc2nocc2C)C1 c1(-n2c(C(C)(CCC3CC3)NC(CCC=C)(C)C)nnn2)ccc2c(c1)CCC2 CN1C(=O)NCC1C(=O)NC1CC(CNC(=O)CC2(O)CCCCC2)C(O)C1 C1(CCCN(C(c2ccccc2)CSC)C)CCOCC1 N1(C(c2cc(OC)no2)=O)CCOC2(CCN(C(=O)CCOC3CCCC3)C2)C1 N1(C(C23C(C)OC(C)(C2)C3)=O)CCC(C2CC2)(CNC(c2ccc[nH]2)=O)C1 N1(C(c2ccc(SC)o2)=O)CCC2(CCN(C(=O)C(C)C3CCC3)C2)C1 N1(C(c2cnccn2)=O)CC2C3CCC(C2C1)N(C(C1(c2ccsc2)CC1)=O)C3 C1(C(N2C(CNC(=O)Cc3ccccc3Cl)CC2)=O)CC12CCSCC2 S(=O)(=O)(c1ccc(Br)c(F)c1)N1CCC2(C(C(=O)Nc3ccncn3)C2)CC1 N1(C(CC=CCC)=O)CCOC(CN(C)C(C2(C#N)CCOC2)=O)C1 C12(C(=O)NCC(C)NC(=O)C(C)(C)NC(c3ccccn3)=O)COCC(C1)OC2 CCCC(C(=O)NC1CC(OCC(=O)NCCN2CCC(C)(C)C2)C1)OC c1(C(C(=O)NC)N(C)Cc2ncc(Cl)n2C)cc2cc(Cl)ccc2o1 N1(CCNC(CC2C(NC(=O)OC(C)(C)C)CCC2)=O)CCCC(N=[N+]=[N-])C1 c1(C(=O)NC(CC)CN(C(=O)CN2CCOCC2)CC)cc2n(n1)CC(O)CO2 C1(NC(C(c2ccccc2)SC)=O)CCS(=O)(=O)C1.c12occc1CS(=O)C2 c1(OC)cc(N2CCC(N(c3cnccn3)C)CC2)nc(C(=O)NC2CCC2)n1 c1(C(N(CCCNC(CC(C)OC)=O)C(C)C)=O)cc(C2CC2)cc(F)c1 C12(C(=O)NC(CC)CNC(=O)Cc3cncc(C)c3)CCCC1NC(=O)C2 C1(C(=O)NC(CCCNC(C(C=C)O)=O)(C)C)CCC(=O)N(C(C)C)C1 c1(CC)n[nH]cc1C(=O)N(CCC(=O)NCCCc1ncc[nH]1)CC1CC1 CCCC(C)CC(=O)NC1(C)CCN(C(=O)C=Cc2cccc(Cl)c2)C1 N1(C(C(C)CN(C)C(c2cnc(O)c(F)c2)=O)=O)Cc2ncsc2C1 N1(C(C2(C)CCC2)=O)CCc2ccccc2C(NC(=O)CSC2CCCC2)C1 c1(CCNC(=O)CC2C=CCCC2)ccc(CNC(C2CC23CCOC3)=O)cc1 C=CCCCC(C(=O)NC(c1ccn(C)c1)C)NC(c1ccc(C#N)cc1)=O N1(C(C(COC)O)=O)CC2CN(C(c3ccnc(OC(C)(C)C)c3)=O)CC2C1 C1(F)(C(N2CC3C(CNC(COCCCC#C)=O)C3C2)=O)C(C)(C)C1(C)C C1(C(=O)NC2(C)CC2)CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1CC1CCCC1 c1(Cc2n(CCOC)c(N3CCN(S(=O)(=O)CC)CC3)nn2)c(F)cccc1F c1(C(=O)NC2C(CC)CN(C(c3csc(O)n3)=O)CC2)noc2cc(F)ccc12 C1(NC(c2c(C)nsc2)=O)CCC(C)N(C(=O)CNC(=O)CCC2CCCC2)C1 N1(C2C(C)(C)C(NC(C3(C)CCCC3O)=O)C2)CCN(c2ccncn2)CC1=O Cc1nc(C(=O)NC(C)(C)CCNC(=O)C(C)C(C)O)ccc1[N+](=O)[O-] c12ccc(cc1F)c1ccc(c(F)c1)o2.C1(OCCC(=O)NC(C=C)=O)CCNC1 c1(C(=O)NC(C(C)C)C(C)NC(c2cn(C)ccc2=O)=O)ccc(O)c(CO)c1 C1(NC(c2c(C(C)=O)ccs2)=O)CCOCC1NC(c1ccc(C(F)F)cn1)=O c1(OC)ncc(C)cc1C(N1CC2(NC(=O)C(C)N(C)C)CC1C2)=O CC1OC(C)C(C)N(C(c2cc(C(F)(F)F)nn2-c2ccccc2)=O)C1 c1(C(=O)NCC2CC(C)N(C(C3CCCC(C)C3)=O)C2)cnc2[nH]nnc2c1 c1(C(=O)NC(C2CCCN(C(CC(C)CF)=O)C2)C)ccnc(Cl)c1F c1(-c2nnc(N3C(CC(C)(C)C)CCC3)n2CCC#N)ccc(S(N)(=O)=O)cc1 c1(OC)ccnc(O)c1C(N1CC=CC(NC(c2nccc(C)n2)=O)C1)=O C1(N(C(C(C2CCC2)OCC)=O)C)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 N1(C(c2c(C)nns2)=O)CCC(C)(CNC(c2cn(CCF)nn2)=O)C1 c1(C(=O)NC2C(C(C)NC(=O)C(C3CCOCC3)=O)CC2)ccc(C(F)F)nc1 c1(C(N2C(C(=O)NC(C)CC(F)(F)F)C=CC2)=O)cc2occc2[nH]1 N1(C(C2CCCC2F)=O)CC2CCCC(C1)N2Cc1c(F)ccc(F)c1O C1(CNC(C2C(CC)CCC2)=O)CCCC12CCN(C(C1C=C1C)=O)CC2 c1(C(=O)OC)nccnc1C(=O)NC(C)CC(C)NC(=O)Cc1cnn(C)c1 c1(C(C)=O)ccc2c(c1)CN(Cc1ccc(-c3ccc(N)cc3Br)o1)CC2 Cc1ncnc(N2CCCC(CO)(NC(=O)CCC3CCCC(=O)N3)C2)c1C#N N1(C(=O)OC(C)(C)C)CCN2C(C1)C2.C1(=CCCCCC)CCCCC1O C1(C(C)C(=O)NCC=CBr)CCN(C(=O)CCc2cccn2C)C1 c1(C(c2nnnn2C(C)(C)CC)NC(c2cccs2)CC)ccc(OC)nc1 c1(C(=O)NC2(CNC(c3c(CC)non3)=O)CCC2)cc2ccc(OC)nc2[nH]1 c1(C(=O)NCC2(NC(=O)C(C)N(C)C)CC(OC)C2)c[nH]c2ncccc12 C1(=CC(CC)C)CCN(C(c2ccc(CC(=O)OC)cc2)C(=O)NC(C)C)CC1 c1(CC)cc(C(N2CCCCC2c2cn(CC3(O)CCC3)nn2)=O)c(C)o1 CC1COc2ccccc2C1OCCN1C(=O)CC(C(=O)Oc2ccccc2)C1 C1(C(N(CCCN(CCO)C(C2CC=CC2)=O)C)=O)CSCN1C(C1CCC1)=O CC1(c2ccccc2)CCN(C(C2CC3CC(Cc4ccccc4)C3C2)=O)CC1 NS(=O)(=O)C1CCC(C(N2CC(NC(c3ccc([N+](=O)[O-])cc3)=O)C2)=O)CC1 C(CCC(C(=O)N(CC)OC)NC(=O)CNC(N)=O)OC N1(C(c2n(CC#N)ncc2)=O)CC2ON=C(CNC(c3ccsc3)=O)C2C1 c1(CC)cc(C(N2CCCCC2CN(C(=O)C2=CCSC2)C)=O)ccc1F c1(CC(C)C)cc(C(=O)NC2CN(C(C3CCO3)=O)C2)no1 c1(C2C(=O)Nc3c(cccc3)N2C)nc2c(s1)CCCC2.C(CCOC)SC C1(CN(C(=O)CSC2CC2)C)CCN(C(=O)CC2CC3CCC2O3)CC1 C(=O)(C(C)CCCC(C)C)NC1CC2CN(C(c3ncc(C)nc3)=O)C(C1)C2 CC1CN(C(C2CCC=CO2)=O)CCC1CNC(c1c(O)cccc1F)=O N1(C(Cn2c(C(C)C)nnn2)=O)CC(Nc2nccc(C(F)F)n2)C(C)(C)C1 C(=O)(C1=CCCCO1)NC1CCC(CCNC(=O)Cc2nc[nH]n2)C1 C1(C(N(OC)Cc2ccccc2)=O)CCN(C(c2ccc(C#N)o2)=O)C1(C)C c1(C(=O)NC2C(NC(c3nc(C)oc3)=O)CCC2)ccc2nncn2c1 c1(C(N(C(C)CS(C)=O)C)=O)n[nH]c2c1CN(C(=O)C1=CCCCC1)C2 Cc1cc([N+](=O)[O-])cc(Cl)c1NC(C1CC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C1)=O Cc1cncc(C)c1C(=O)NC(Cn1cncn1)C(=O)NCC1CC12CC2(F)F C1(CC(N2CC(C)(ON(CCCOC)C(=O)COC)C2)=O)CCCC(C)O1 C1(C(=O)NCCc2c(C)noc2)(CNC(=O)CCC2CCCCO2)CC12CCC2 c1(OC)cccc(C(C)C(=O)NC(C)C(C)NC(=O)CSC)c1 C(=O)(C1CCCc2nn[nH]c21)NC1C(C)N(C(=O)COCCN(C)C)CCC1 N1(C(c2c(CC)cc(Cl)cc2)=O)CC2(CC(NC(=O)C(C)(Cl)Cl)CO2)C1 N(C(=NCCc1cccs1)NCc1cnc(Br)s1)CC1CCCC(C)C1 C1(C(=O)NCC(C)NC(c2cocn2)=O)CCCCC1P(C)(C)=O C(CCCCC(=O)N1CC(O)CC1(C)C)N(C(C1C(CC)CCO1)=O)C c1(OC)ccc(-n2nnnc2C2(NCCOCCO)CCCC2C(C)(C)C)cc1 C(=O)(C(C)(C)CO)N1CC(N(C)C(C2CCC(C(F)(F)F)O2)=O)C1 N1(C(COCCC)=O)CC(O)C(O)C1CNC(=O)CC1OC(C)(C)OC1=O c1(C(N2CCC2CNC(C2(C3CC3)CC2)=O)=O)cc(Cl)ccc1[N+](=O)[O-] S(=O)(=O)(c1ccccc1Br)Nc1c(C(CC(C(C)(C)C)=O)=O)scc1 C(CCF)(C(=O)Nc1ccc(CO)nc1)NC(C1CC=CC(O)C1)=O C1(C(N(CC(C)NC(COC)=O)C)=O)(NS(CC)(=O)=O)CCSCC1 C1(C(=O)OCCC#CC)Cc2ccsc2CN1C(=O)NC(C)(C)C C1(NC(COCC(=C)C)=O)CCN(C(C23CCCC2C3(F)F)=O)C12CCC2 c1(C(=O)NC(CNC(COCCOCC#C)=O)CO)c(F)cc(F)cc1Cl c1(CCC(=O)N(CCN(C)CC2CCN(CC)C2)C)ccc(O)nc1 c1(CC(=O)NC2CC(CCNC(c3cn(CCC)nn3)=O)C2)ccc(Cl)c(F)c1 N1(C(C(C=C)OC)=O)CC(C(=O)NCC2(N(C)C)CCC2)C(C2CC2)C1 N1(C(C(C(C)C)N(C)C)=O)CCCOC(CNC(C2CCC3(CC3)C2)=O)C1 CC1CCCC(C)N1C(=O)Cn1cc(-c2ccc(F)cc2)nn1.C(C(=O)O)N CCC(C)C(C(=O)N(CCCCCNC(c1ccc(F)cc1)=O)C)OC C(=O)(N1CC(C)(O)CO1)C1(CNC(C(C)(C2(C)CC2)NC(C)=O)=O)CC1 C1(CCC)C(=O)NCCN1C(C1CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1)=O N1(C(CC2CN(C)C2)=O)CC(CNC(=O)CCn2cnnn2)CC1(C)C C=CCC(C)C(=O)NC(C)C(C1CCCCC1)NC(=O)CCCNC(=O)C1CC1 N1(C(c2ccc(-c3cccc(F)c3)cc2)=O)CCC2(C1)CN(C(C1CC1F)=O)C2 N1(C(c2cc(C)c(F)cc2)=O)CCN(C(c2cc([N+](=O)[O-])sn2)=O)CC(O)C1 CCCCC(O)C(C)C(=O)N1CCC(C(=O)NC(C)C(C)SC)(CO)C1 C1(NC(=O)COc2ccc(F)nc2)CCC12CCN(C(C1CCCO1)=O)CC2 c1(OC(COCCC)NC(=O)CC)cccc(C(=O)NCC2CC2)c1 c1(C(=O)NCC(=O)NCc2nc[nH]n2)cc(CO)cc(F)c1.C12CC(C1)C(=O)N2 c1(CN(c2cc(N(C)Cc3ccns3)ncn2)C)cccc(Cl)c1Cl C(CCCC(C)NC(=O)CC=O)N.C(=O)(CC(C)(C)OC)SCCN(CC)CC C1(C(=O)NCC2CN(C(=O)CN3CCCNS3(=O)=O)C2)CC2(CCC2)CCO1 O=C(N=c1c(Br)c[nH]cc1I)C1CC(O)CCN1S(=O)(=O)C1CC2CCC1C2 c1(C(=O)NC2C(NC(C(C)CC3CC3)=O)CCOC2)coc2ccc(F)cc12 C1(NC(c2cnc(C)nc2)=O)CN(C(c2cccc(Br)c2N)=O)C(C)(C)C1 c1(C(=O)OC2CC2)cccc(S(=O)(=O)NC2CCC2n2ccnc2)c1 C12(CNC(C3C(OCC)C3)=O)CC1CN(C(=O)COCc1nc(C)no1)C2 N1(C(CNS(NC)(=O)=O)=O)CC2CN(C(=O)C=CC3CC3)CC2C1 Cc1nc(C(F)(F)F)sc1CC(=O)N(CCCN(C(=O)CC1CCCC1C)C)C Cc1ccc(F)c(C(=O)NC(CC(C)C)C(=O)N(C2CCOC2)CCF)c1 C=C(C)CC(C(=O)NCCc1cnn(C)c1C)NC(=O)CNc1ccccn1 S(=O)(=O)(c1c(C)cc(C)cc1C)NCC(=O)NC(CC#C)C c1(C(=O)NCC(CNC(CCC#C)=O)F)cc(F)ccc1-n1ccnc1 c1(C(=O)NC(CNC(CC(CC)C)=O)(C)C(C)C)ccc(C)c(N)c1 CC1(C)CCCCC1n1cc(C2CN3CCC2(C(=O)O)C3)nn1 C(CCCC(=O)N1CCC(F)(CNC(C2(Cl)CC2(C)C)=O)C1)N(C(C)=O)C N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NC3(CO)CCOC3)C2)C1 CC1(C)CC(=O)NCC1C(=O)NC1(CF)CN(C(=O)CCCCN=[N+]=[N-])C1 CC(O)C(F)(F)C(=O)N(C)CC1CN(C(C2CCC(C(F)(F)F)CC2)=O)C1 N1(C(CC2CC(C)C2)=O)CCC(C)(CC(=O)N(CC(C)(C)C)C2CC2)C1 C1(N(C)C(c2cnn(-c3ccccc3)c2F)=O)CCCN(C(=O)CC#N)C1 c1(C(=O)NCCCCCNC(Cc2cncc(C)c2)=O)cc(F)c(C#N)c(F)c1 C1(N)(C(=O)NC(C(=O)OCC)CSC)CCOCC1(C)C C#Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(C)(C)C2)=O)ccc1C Cc1ccc(C(N)=O)cc1S(=O)(=O)NCC1CCN(C(=O)C(C)C)CC1 C12(NC(C(CCN(C)C)O)=O)CCCC1CN(C(=O)C=Cc1ccccc1F)C2 c1(OC)cc(C(=O)NCC(C)N(C(=O)CC(C)(F)F)C)ccc1OCCN(C)C N1(CC)CCC(NC(=O)C(CC2CCC2)NC(C2CN(C(C)=O)C2)=O)C1 CC(C)C(C(=O)NC1CCN(C(C2(C)CCC2)=O)CC1F)C(C)C C(=O)(C1COc2ccccc21)N1CCCC2(CN(C(=O)Cc3ccc(Cl)s3)C2)C1 C1(CNC(CC(C=C)CC)=O)CN(C(C2CC(CC(F)F)C2)=O)CCC12CCC2 N1(C(C2(SC)CC(=O)C2)=O)C2CCC1CC(C(N1CC(C)(C(N)=O)C1)=O)C2 C(=O)(C1CC(=O)c2ccccc21)N1CCC(F)(C(=O)OC(C)(C)C)C1 N1(C(CSCCN(C)C)=O)CCC(C(CO)NC(=O)CCc2ccon2)CC1 CS(=O)(=NC(=O)CCn1cc(Br)cn1)c1ccccc1Cl CC1CC(CNCc2ccnc(-c3ccccc3C(=O)O)c2)CC(C)O1 c1(C(=O)NCc2ccc(-c3cc[nH]c3)nc2)ccc(O)cc1Cl CC1COCC(C(=O)NC2CC(O)(CNC(c3cccn3C3CC3)=O)C2)O1 C1(C(C)(C)C)CCN(C(c2cc[nH]n2)=O)C(CNC(C2CCCOCC2)=O)C1 N1(C(C(CCO)N(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2cnco2)=O)C1 Nc1ncc(C(=O)NCCOC2CCN(C(=O)C=CC3CCOC3)C2)cc1Br c1(OC)cnccc1C(N1CCOCC1C(=O)NCCOCC1CCOC1)=O CC(Cc1cnn(C)c1)C(=O)NC1CN(C(=O)COc2ccsn2)C1 N1(C(CNC(C(C)(C)OC(C)C)=O)=O)CCC(O)C(C)(C)C1 C1(O)(C(=O)NC2CC3(CC(NC(c4scc(C)c4C)=O)C3)C2)CCCC(C)(C)C1 N1(C(C23CCN(C(c4cc(C)on4)=O)CC2C3)=O)CCC(C)(C#N)CC1 C1(CCNC(c2ncn(CC)c2)=O)C(C)CCCN1C(=O)C1=COCCC1 c1(OC)ccccc1NS(=O)(=O)CCC1CCN(C(c2cscn2)=O)CC1 c1(C(C)C)cnc2c(c1)C1CCC(NCCCCC3(C#N)CCC3)C21 c1(C(=O)NCCC2N(C(C=CC(CC)=CC)=O)CCC2)ccc2cc[nH]c2c1F c1(N2CCN(C(C34CC(CCC)(C3)C4)=O)C(C)CC2)nc(Cl)nc2c1CCOC2 C(CN=c1[nH]c2ccccc2s1)N(C(C1N(CCC)CCCC1)=O)C N(C1COc2ccc(F)cc21)C(N(c1c(C)cccc1)CCO)=O C(=O)(CC(F)(F)C(F)F)N1CC(C(=O)NCc2nonc2C)(OC)C1.N C1(CNC(CC=CCNC(CCCOC)=O)=O)COCC(C)O1 Cc1cc(CCNC(=O)C(F)CN(C(=O)CC2CC(=O)C2)C)on1 C1(C(=O)NC2CCN(C(c3c[nH]c(=N)o3)=O)C2)CCC(c2ccccc2)CC1 O(N=C1CCCCCC1)CC(N1CC(CC=C)(NC(=O)CSCC(F)F)C1)=O C1(C(N2C(C(=O)NCc3ccccn3)CC(O)C2)=O)CCCC2(CC2)C1 C1(C(=O)NCC(C)N(C)C)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C N1(C(Cc2cccc(OC)c2)=O)CCc2[nH]nc(CNC(=O)C(C)NC(C)=O)c2C1 N1(C(c2c(C)c[nH]n2)=O)CC(NC(=O)Cn2nnc(=N)[nH]2)C2(CCC2)C1 N1(C(c2ncn(C)c(=O)c2)=O)CC2CC(C1)N2C(=O)CC1CCCC2CC12 N1(C(=O)Cc2csc(O)n2)CCCCC1C1CCN(Cc2cnccn2)C1 C(=O)(C(F)C(F)(F)F)N1CCC(OCCNC(=O)Cn2nnc(=O)[nH]2)CC1 c1(NC(C2(NC(C(C)CCN(C)C)=O)CC(F)C2)=O)cnc2[nH]ncc2c1 C12(CNC(C3(c4cc(C)no4)CC3)=O)CC(CN1C(c1c[nH]c(=N)s1)=O)C2 C1(CCC)CN(C(C2CN(CC)CCO2)=O)CC1NC(c1cccc(N)n1)=O Cc1nc2ccc(C(=O)NC3CC4CC3N(C(=O)CC35CCCC3C5)C4)cc2o1 c1(NC(CCc2ccc(C(=O)OC)[nH]2)=O)nc(OC)ccc1Cl N1(CC(c2ccccc2Cl)(C)O)CCC(C#N)(C(=O)O)CC1 N1(C(c2c(C(C)(C)N)noc2)=O)CC(=O)N2CCCCC2C1 c1(C(=O)NCCN(C(C(C)SC)=O)CC(C)O)cc2c(cn1)OCCO2 Cc1c(C(=O)NC(c2cccc(C(=O)O)c2)CO)sc2ccccc12 N1(C(=O)NCC(N2CCCC2)C)CCN(C)C(CO)C1 c1(N(C)CC2CCN(C(c3ccccc3)=O)C2)ncnc2c1ncn2C c1(C(=O)NC(CCOC)CNC(=O)CC(F)(F)Cl)ccc(N=[N+]=[N-])cn1 CC(CS(=O)(=O)N1CCC(O)C(C(N2CCCC(O)CC2)=O)C1)C(C)(F)F Cc1ccc(C(=O)NCC2(C(=O)NCC3NC(=O)NC3=O)CCCC2)nc1 Cc1nncc(C(=O)NC2CC(F)(F)CC2NC(C2CCSC2)=O)c1C N1(C(C(=O)NCc2ccccc2)C2CCSC2)CCn2c(cc3c(Cl)cccc23)C1 c1(OC)ccc(C(=O)NCC2C(C)CCN2C(c2coc(C(C)(C)C)n2)=O)nn1 C1(C(N2CC(CC(=O)NCC3CC(OC)C3)(OCC)C2)=O)CC12CCCC2 c1(C(C)NC(=O)NCC2CCC(CO)O2)cccc(N2CCCC2)c1 Cc1nc(C(=O)NC(C)CC2CN(C(=O)OC(C)(C)C)C2)ccc1C(F)F c1(CC(C)NC(=O)C=CCNC(C2CC2F)=O)cccs1 N1(C(Cc2cc(OCC)no2)=O)CCS(=O)(=O)CC1C1CC1 C1(C(=O)NCC(CN(C(c2ccc(SC)s2)=O)C)C)CCCC2(C1)CC2(F)F c1(OC(C)C)cccc(NCCC(C(C)C)NC(c2cnc(Cl)cn2)=O)c1[N+](=O)[O-] N1(C(C(C)(C)C#N)=O)CC2CC1CC2CNC(=O)CSc1cccs1 c1(C(N(CCNC(C(C#C)(C)C)=O)CCC)=O)cc(O)ccc1OCC(F)F C(C(F)(F)C(=O)N1CCN(C(=O)C(=O)Nc2ccccc2)CC1)N(C)C c1(C(=O)NC2(C)CCN(C(c3nnn(C)n3)=O)C2)cccc(F)c1Br C1(NC(CC(CC)OC)=O)CCCCC12CCN(C(c1c[nH]nc1OC)=O)CC2 N1(C(c2sccc2Cl)=O)CC(CO)C2(C1)CN(C(c1csc(O)n1)=O)C2 C(=O)(C(CCC)C(C)C)NCC1(F)CCCN(C(COCC(=C)C)=O)C1 Cc1ccccc1C(=O)NCc1nc(C(=O)NCCC2CCSC2)c(C)o1 CC1CN(C(=O)C2=CCCS2)CCC1NC(c1cnc(N(C)C)c(Cl)c1)=O Cc1csc2ncc(C(=O)NCc3cccc(N)c3F)n12.C12CCCN1C2=O C12(C(=O)Nc3ccc(C)cc3CO)COCC1CN(C(=O)CCC(CF)CF)C2 c1(C(C(=O)N(CC(C)O)CCNC(CCC(=O)OC)=O)C)cc2ccccc2o1 N1(CC)CC(CNC(C2(C(=O)NCC3(C(=O)NC)CC3)CC2)=O)CC1C c1(C(N2CCN(C(CS(CC)=O)=O)CC2CCO)=O)cc2c([nH]1)CCOC2 C1(CNC(C(CC)F)=O)CCCCCN1C(=O)CSc1ccc(OC)cc1 C(=O)(C1=C(C#N)CCC1)NC(C(=O)NC(C)Cc1ccoc1)CCF N1(C(c2c(C)noc2N)=O)C2CCC1CC(NC(C1CCC3(CCC3)CC1)=O)C2 N#CC1(C(N2CCC(O)(CNC(c3cc(Cl)c(Cl)s3)=O)C2)=O)CC2(CC2)C1 Cc1cc(NC(=O)CCC2CCN(C(C3CC3C#N)=O)C2)cc(C)c1C Nc1ccnc(C(N2C3CCC2C(NC(=O)Cn2nccn2)C3)=O)c1Cl Cc1nc2c(C(=O)NCCNC(=O)Cc3ccc(C)c([N+](=O)[O-])c3)ccnc2[nH]1 CC1=NOC(=O)C1CC(=O)NC1CCC1NC(c1ccncc1OC(C)C)=O c1(CN(C(C=C(C)CNC(=O)CC(C)N(C)C)=O)C)nocc1C N1(C(C(CO)OC)=O)CC23CCCCC2(C1)CN(C(c1ccc(Cl)o1)=O)C3 CC(C)C(O)C(=O)NCC12CC1CN(C(c1ccc(CO)cn1)=O)C2 C1(C(=O)NCC2CCCN(C(=O)Cn3cncn3)CC2)Cc2cccc(F)c2O1 C1(C(c2nc(C)c(C)[nH]2)c2nnn[nH]2)CCCCC1NCc1cccs1.CO CC(C(O)C(F)F)NC(C1(NC(=O)C#CC2CC2)CC(F)C1)=O N1(C(C2C(C)(C)C(NC(c3cccc(CO)c3)=O)C2)=O)CCCCCCC1 c1(C(N2CC(NC(C(CC)(C)CO)=O)CC2(C)C)=O)c[nH]c2cc(F)c(F)cc12 C12(CNC(CN(C(C(n3ncc(C)c3)C)=O)CC3CC3)=O)CCCC(CO1)C2 Cc1ccn(C(C)C(=O)NC2CCOC2C(=O)NCC(O)CNC(=O)C2CC2)n1 CCC(CC(=O)NCC1CCCN(CC(=O)NCCCC(C)C)C1)C(C)(C)C c1(C(=O)NCC(CC)NC(C(C2CCC2)OCC)=O)oc(Br)cc1C CC1(CNC(=O)C(CCl)NC(N)=O)CCCN(C(=O)CC23COCC(C2)C3)C1 C1(O)(C(=O)NCC2(O)CCN(C(CC3(C(=C)F)CCC3)=O)C2)CN2CCC1CC2 c1(NC(C(=O)N(C)CC2CCC(C)C2)=O)cccc(Br)c1F c1(OCC(=O)NCC(CCOC)NC(c2ncoc2C(C)C)=O)ccc(F)nc1 C(C)(C)(CC(=O)NCC(C)(O)CSC)NC(C(CC)SC)=O C1(NC(CCSC)=O)CCC(C)N(C(c2cnc(N3CCCS3(=O)=O)s2)=O)C1 C1(C(C(=O)NCCCSCC)N(CCCC)C)C2CCCCC12 c1(N2CCC(NCC(C(C)C)NC(=O)C3=CCOC3)C2)ncccc1C(F)(F)F N1(C(COCCCOC)=O)CCCC12CCCN(C(c1cc(C)oc1C)=O)C2 c1(NCCC2CCN(C)C2)ccc(C(F)(F)F)cc1S(=O)(=O)N1CC(F)(CF)C1 N1(C(C2(COC)CC(=C)C2)=O)CCCCC1C1CCN(c2nnnn2C)C1 c1(C(=O)NCCOC2CCN(C(CC=CC=C)=O)C2)cc2ncccc2cc1Cl N1(C(CCNC(=O)NC)=O)CCN(C(C2CCN(C)C2)=O)CC1CS(C)(=O)=O Cn1cc(C(F)(F)C(=O)NC2CCC2NC(=O)CC2CC=CC2)cn1 C#CCC(CC#C)C(=O)NC1CN(C(=O)C(n2ccc(C)n2)C)CC1C1CC1 C1(C(=O)NCC(C)NC(c2c(C)noc2C(C)C)=O)CC(c2ccncc2)=NO1 c1(C(=O)NC(CN(C(c2c(C)scc2)=O)C)C)c[nH]c(=O)cn1 C1(C(C)C)CN(C(=O)CN2CC(=O)N(C)C2=O)CCN1C(=O)CC1CNC(=O)O1 Cc1cc(N)c(C(N2CCN(C(=O)Cn3cnnc3O)CC2CO)=O)cc1C C1(NC(c2ccc(CC)o2)=O)CC(F)CN(C(C2CC2(Cl)Cl)=O)C1 C1(C(N2CC(O)(CNC(C3(CCC=C)CC3)=O)C2)=O)COc2cc(F)ccc2O1 C(CC1CCC1)(C(=O)NC1CCC2CC12)NC(C(C)=C1CCC1)=O c1(OCS(N)=O)ccc(C2(CN3CCN(Nc4ccc(Cl)cc4)CC3)CC2)cc1 n1(CC)ccnc1C(=O)N(CC(=O)N(CC(Cl)Cl)C)C(C)C C1(C(N2CCCCC(NC(c3c(C)occ3)=O)C2)=O)Cc2ccccc2C1(C)C C1(C(c2nnnn2CCCCCO)NCC(C)(C)OC)C2CC3CC(C2)CC1C3 C(=O)(C#CC1CCCOC1)NC1(CO)CCN(C(c2nnc(C)s2)=O)CC1 N1(C(CC2CC(OC)C2)=O)CCN(C(=O)C(C)C(=O)N2CCOCC2)C(C)C1 N1(C(=O)CC2CCCC3CC23)CC2(C(N3CCC(N4CCC4)C3)=O)CC1CO2 C1(C(=O)NCC(CC)O)C2CCCC2CN1C(C1CCC1C)=O CC(C)C(C)(O)C(=O)NC(C)CCC(=O)OC(C)(C)C C1(SCC(=O)NC2CC2NC(c2ccc(C(F)(F)F)o2)=O)CCOCC1.CCCC C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CC2CCOC2(C)C)CCC1(C)C N1(C(c2c(C(F)(F)F)oc(C)c2C)=O)CCN(C(=O)CC2CCCC2)CC1C CCC(CC(=O)N1CC(C2CN(C(c3c(CC)nc(C)n3C)=O)C2)C1)C(C)C c1(C(=O)NCCCCN(C(Cn2c(C)cc(C(F)F)n2)=O)C)ccc(Cl)cc1N Cc1cc(N2CCC3(C)C(C2)C3(Cl)Cl)nc(=NCCN2CCOC3(CCC3)C2)[nH]1 c1(OC)ccccc1OCC(=O)NCC1CCN(C(c2ccnnc2Cl)=O)C1 c1(C2N(C(c3c(CC)oc(C)c3)=O)CCC2)nc2cnccc2[nH]1 N1(CN2C(=O)CC(C(=O)OCCOC(CC=C)=O)C2)CCCC(C2(OC)CC2)C1 C1(CNC(C2(NC(C3C=C(C)CS3)=O)CC2C)=O)CC12CCOCC2 Cn1cc(-c2ncc(C(=O)NCC3CCCC3NC(c3cnc(O)o3)=O)s2)cn1 N1(C(=O)CCc2ccccn2)CCOC2(CCN(C(C3CC3F)=O)C2)C1 C1(NC(c2c(CC)nc(=N)[nH]c2)=O)COC2(C1)CN(C(=O)C1=C(Cl)CCCC1)C2 CCCC(C)C(=O)NC1(C)CN(C(C23CCC2C3)=O)C1 N1(C(C(CC)SC)=O)CCC=CC1C(N1CC(C#N)(OC)C1)=O N1(C(c2c(Cl)cn(CC)n2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)C(C)C)C2 Cc1cccnc1C(=O)NCCC(C(C)C)NC(c1ncnn1C)=O CC1CC(C)N(C(c2ccnnc2S)=O)CCN1C(c1cnc(O)n(C)c1=O)=O C(=O)(C(C)N=[N+]=[N-])N(CCC(=O)N(CC(O)CO)C)C(C)C CCCCCCC(C)CC(=O)NC1CN(C(C2CCCO2)=O)CCC12CCC2 c1(OC)ccc(C(N2CC(NC(=O)CCC3CCCO3)C2)=O)c(F)c1 N1(C(CC(C)C)=O)CCCC(NC(c2cccc3ccsc23)=O)CCC1 c1(C(N2CCOC(c3nc(C(=O)OC)cs3)C2)C(=O)NCC)cccc(CO)c1 c1(C(N2CCC(C)(NC(C(CCCCC)O)=O)C2)=O)cnc2ccccc2c1 N1(C(c2ccccc2C(F)F)=O)CC(CO)C2(C1)CN(C(C1CCCCO1)=O)C2 C1(C(C)C)CCN(C(=O)Cc2ccc(Cl)s2)C(CNC(=O)C(=O)NCC(F)F)C1 Cc1cnn(CC(=O)N(C)CC2CN(C(c3cnc(CC(C)C)s3)=O)C2)c1 c1(NC(C2CCC(NC(c3ccc(C(F)(F)F)cc3)=O)CC2)=O)cnccc1Br C1(CNC(C2C(C)=CCS2)=O)CCCCN(C(=O)CC2CCCO2)C1 N1(C(C=NOC)=O)CCC(C)(C)C(NC(=O)COc2ccc(Br)cc2)C1 N1(C(C2(COC)CC2)=O)CCC(C2CCCN(C(=O)Cc3sccc3C)C2)C1 C1(CNC(C(F)=C(C)C)=O)CCN(C(=O)CCn2ccc(C)n2)CC1CO c1(C(=O)NCC(C)NC(C2CCCCN2C2CCCC2)=O)c[nH]c2cccnc12 n1(CC(=O)N(C)CCNC(=O)CC2CC2)ncnn1 CN1N=C(CC(=O)N2CCCC(NC(C3(n4nccn4)CC3)=O)C(F)C2)CC1=O C1(C(N2C(CCC=C)CCC2)=O)CN(CC2CCC(CNC(C)=O)O2)CCO1 c1(OC)ccc(CN=C(NCC2(CS(C)(=O)=O)CCC2)NCC(C)(C)C)cc1 N1(C(C(=O)NCC(=O)N(c2ccc(F)cc2)C)=O)CCC2(CCCNC2)C1 C(CN=C(NCc1ccc(C)n1C)NC1CCCC(F)(F)C1)SC Cc1ccc(C(N2CCCCC2CCC(=O)NC(C)CCC2CC2)=O)nc1 c1(CCC(=O)NCC2C(NC(C3(CCOC)CC3)=O)CC2)ccc(O)nn1 c1(C(=O)NC2C(C)CCN(C(=O)C(C)(C)C)C2)cc(F)cc2c1C(=O)CC2 N1(C(CC(C)SC)=O)CCC(C2CCN(C(=O)CC3=NN(C)C(=O)C3)CC2)C1 CCC(CC)C(C(=O)NCC1(C(=O)N(C2(CO)CC2)C)CC12CCC2)OC C(CC1=CCN(C(C2CN(C)CC2C)=O)CC1)NC(C(C)(C)OC)=O CC1C(NC(c2cn(CC(F)F)cn2)=O)CCN1C(C1CCOCC1)=O N1(C(C=C(CC)CC)=O)CCC2(CC1)CN(C(C1CCCC(C(N)=O)CC1)=O)C2 c1(C(N(C(CC(=O)N(CC#C)CCF)CC)CC)=O)c[nH]c2cccnc12 S(=O)(=O)(CC(C)CC)N1CCN(Cc2cn(CCCC)nn2)CC1 C1(O)(CNC(N(CCCCC)Cc2ccc(F)cc2)=O)CCS(=O)(=O)C1 Nc1c(C(N2CCC(CNC(C3(C(N)=O)CC3)=O)C2)=O)sc2ccccc12 C1(C(N(C)Cc2ccc(C)cc2)=O)CC(C)CCN1C(=O)CC1CCSC1 C1(CNC(CCNC(C(c2ccn(C)n2)C)=O)=O)CCCCC1CO c1(C(C(=O)C(Cc2cc[nH]n2)NC(=O)C2CC2)=O)cc(F)ccc1O.C1(N)(CF)CC1 N1(C(c2cncc(Br)c2)C(=O)Nc2ccc(F)cc2)CCn2ncnc2C1 c1(C(=O)NC(C2CN(C(=O)CN3CCCC3=O)C2)C)cc(-c2ccccc2)cs1 O=C1CCC(C(=O)NCC2(O)CCN(C(=O)CSCc3ccccc3)C2)CN1 c1(C(=O)NCC2C(CNC(C(CC)O)=O)C2)cccc(OCCO)n1 C1(NC(=O)CCSC(F)(F)F)CC12CC(NC(c1c[nH]nc1F)=O)C2 N1(C(c2cn(C)nc2)=O)CC2C3CCC(C2C1)N(C(c1ccc(S)cc1)=O)C3 C1(NC(=O)NC(c2ccccc2)CN(C)C(=O)OC(C)(C)C)(COCC)CCSC1.CC [N-]=[N+]=Nc1cc(C(N2CC(C(F)F)C3(CC3)C2)=O)ccn1 N1(C(c2c(CC)csc2)=O)CCN(C(c2cc(OC)cs2)=O)C(COC)C1 C1(CC(=O)NC(C)CNC(=O)Cc2nc(=N)[nH][nH]2)CCCCC1F c1(-c2ccc(CN3CCCC(C)(C(=O)OC)CC3)s2)ccc2ccccc2c1 C(=O)(CCCS(C)(=O)=O)NCC(C)(CNC(C1CCCCS1)=O)OC O=C1CCc2nc(N3CC4CCC3C(NC(C3CCCC5(CC5)C3)=O)C4)ccc21 C(C(C)C(=O)NCC1CCC(=O)O1)NC(=O)NC1CC(SC)C1 C=CCCC(CC(C)C)C(=O)NC1(CCNC(C2CCN(CC)C2)=O)CC1 C12CCCC1NCC2.C(CCN(C)C)N(CCN(C)C)C=O C(=O)(C1CNC(=O)c2ccnn21)N1CCC(C(C)NC(c2cnns2)=O)CC1 Cc1ncc(Cl)cc1C(=O)NCC(F)CNC(c1cnn(-c2ccncc2)c1)=O N1(Cc2cccc(CNC(C(C)OCC)=O)c2)CCN(c2ccccc2)CC1 c1(C(N2CC(O)(CCNC(C(CC)(C)O)=O)C2)=O)cnc2c(c1)c(C)nn2C C1(NC(CCC(C)=O)=O)CC2CCC(C1)N2Cc1cc(I)c(C)cn1 c1(OC(C)C(=O)NCC2CCN2C(=O)CN(c2cnccn2)C)cccc(F)c1 c1(C(N2CCC(CCOC)(NC(COCC)=O)C2)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NC2(C)CCN(C(CC=CC=C)=O)C2)cc2c(Br)cccn2n1 c1(C(c2cccc(Cl)c2)CCc2cn(CC(=O)N(C)CCO)nn2)cccc(I)c1 c1(CN(CC(=Cc2ccco2)C)C)ccc(Cl)c(C)c1 CCC(CC)(CO)C(=O)NC1CCC1NC(c1ncc2[nH]ncc2n1)=O N1(C(CCC=C=C)=O)CC(NC(=O)C(N2CCNC2=O)C)C2(CCC2)C1 CC1=C(C(=O)NC2CCC(NC(=O)Cc3n[nH]cc3Br)C2)C(=O)OC1(C)C C1(C(N2CCC(N(C(=O)Cc3nnc(C)o3)CC)C2)=O)OCCOC1(C)C CCCC(C)CC(=O)N1CC2CC2C1CNC(=O)Cc1ccccc1OCC c1(C(=O)NC(CCCC)CNC(=O)C=CCOC)cnc(OC)c(Cl)c1 c1(C(N2CC3CCC(C2)N3C(=O)C=C2CCCCC2)=O)nc(Br)cn2ccnc12 N1(C(c2c(C)[nH]cc2)=O)CCc2ccccc2C(NC(=O)C2=CC3CCC2C3)C1 Nc1[nH]c(=NCCOC(=N)O)[nH]c(=NC2CCC(F)(F)C2)c1Br C1(CNC(NC(CC)C)=NCC2CCC3(CCC3)OC2)CC2(CO1)CC(F)(F)C2 C1(CNC(C2CC(SC)C2)=O)CC2CCCCC2N1C(C1CNC(=O)C1)=O C(CN=c1nc(C)c([N+](=O)[O-])c[nH]1)NC(C1(C)C(CC)CCC1)=O c1(C(N2CCCCC(CO)C2)=O)cn2ccccc2n1 c1(C(N(CCC(C)NC(=O)CO)C)=O)cncc(-c2ccc(F)cc2)c1 c1(OC)cc(C(=O)N(CC(C)NC(C2(C)CCCNC2=O)=O)C)cc(Cl)c1 CN1CCN(C(c2cccnc2N)=O)CC1CNC(=O)C#CC1(C)CC1 CCCC(CC)C(=O)N1CCCC1C1(C(=O)NC2CCCC(C)(C)C2)CC1 c1(OC)nc(N2CCOC(CCNC(c3ccn(CCO)c3C)=O)C2)cc(C)n1 CCCC(CCCO)C(=O)N1CCC2(C1)CN(C(c1cnn(C(F)(F)F)c1)=O)C2 n1(CC(=O)NC(C)C=CC(=O)N(CC2CC2)CC2CC2)ncnn1 c1(C(=O)NCC(CC)NC(c2ccc(COC)s2)=O)c[nH]c2nccc(Cl)c12 c1(C(N)=O)ccc(CCNC2CCCN(CCN)C2)cc1 N1(C(c2cnc(Cl)s2)=O)CC2CC(C1)N2C(c1cnn2ccsc12)=O c1(C(N2CCC(N(C(C(COC(C)C)(C)C)=O)C)C2)=O)n[nH]c2c(C)cccc12 C1(C(N(C2CCSC2)C)=O)CC(C)(C)CCN1C(=O)CCn1cnnn1 N1(C(C2CN(C)C(=O)N2)=O)CCC2(CCCN(C(C3CC(Cl)(Cl)C3)=O)C2)C1 C1(C(=O)NC2C(NC(COCCC(C)C)=O)CCC2)CCCCN(C)C1=O CN1CCC(C)(C(N2CC(CNC(=O)C(F)CC3CCCC3)C2)=O)C1=O N1(C(C2CC3C=CC2C3)C(=O)NCCC2CC2)CCCN2CCCC2C1 C(CCc1ccc(Br)cc1)(C(=O)NC(C)C)N(c1ccc(C(N)=O)cc1)CC Cc1ccc(S(=O)(=O)NC2CC2c2ccc(O)cc2)cc1C Cc1[nH]c(C#N)cc1C(=O)NC(C(=O)NC1C=CCCCC1)C(C)(C)O CCC(C)CC(=O)NCc1ncoc1CCNC(C1CC(C)C(C(=O)OC)O1)=O N1(C(C=CC(CC)C)=O)CCCC(O)(CNC(c2ccsc2)=O)CC1 c1(C(N2CCC(F)(CNC(c3c(C)cco3)=O)CC2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(CCS(=O)(=O)c1ccccc1)NCC1C(C)CN(C(=O)C(=O)NC2CC2)C1 C=C(C)C1OCCCC1C(=O)NCC1CCCN(C(c2cnn(CC)c2)=O)C1 Cc1oncc1C(=O)NCC(=O)NC1CC1CNC(C1CCNC1=O)=O c1(C(C)C(=O)N(C(C)(C)CN(C(=O)C(C)c2ncco2)C)CCO)ccn(C)c1 C1(CC(=O)NCCOC)CCCN1C(c1ccsc1Cl)=O c1(NC(=O)C(N2CCC(Oc3ccccc3)C2)=O)cc(Cl)ncc1Cl c1(C(C)NC(=O)CCn2cc(-c3cc[nH]n3)nn2)cccnc1Cl Cc1cc(Br)cc2cc(C(N3CCCC3CNC(C3(N(C)C)CC3)=O)=O)oc12 CCN=c1[nH]cc(C(=O)N(C)CC2CCN(C(C3CC3F)=O)C2)s1 Cc1coc(C)c1C(N1CCN(C(N2CCN(C(=O)C(C)N(C)C)CC2)=O)CC1)=O CN1CC2(CCN(C(C3CCN(Cc4csc(Br)c4)C3)=O)CC2)C1 CCC(F)(F)CC(=O)NC1COCC1CC(=O)NCCCSC C1(CNC(=NCC)NCc2ccco2)CCC2(CCC2)C1O N1(C(CC2N(C(=O)Cc3ccc(O)cc3)C3C2CCC3)=O)CCC(F)(F)CC1 Cc1cc(Cl)c(C(N2CC(NC(c3coc(C(F)F)n3)=O)CC2C)=O)cn1 N12CCC3C(CCCN3C(=O)CC1=O)C2.c1(OCCOC)ccc2occc2c1 c1(C(N2CCC(C)(CNC(c3cc(N)cc(N)c3)=O)C2)=O)ccc2nsnc2c1 C1(CNC(c2n[nH]c(C)c2O)=O)CC2(C1)CN(C(=O)CCCN1CCCC1)C2 C1(CN(C)C(C2CN(C3COC3)C2)=O)CC2(CO1)CN(C(=O)CNS(C)(=O)=O)C2 c1(C(N2C(CNC(Cc3c(C)nn(C)c3)=O)CC(O)C2)=O)nccc2[nH]ccc12 OCCC(N=c1nc2sccc2c(NCc2ccc(Br)s2)[nH]1)c1ccco1 c1(OC)ccc(C(N2CCC(C(=O)NCc3cc(C)ccn3)CC2)=O)c(Cl)n1 Cc1nnccc1C(=O)NC(C)CCCNC(C1COC(=O)N1C)=O C1(NC(c2ccc(Cl)c(F)c2)=O)CC2CC1CN(C(=O)C(F)(F)CO)C2 C#CCC(CC(=O)N1CCCCC1CCO)NC(=O)CCc1nc[nH]n1 N1(C(c2c(C)ocn2)=O)CC2CCC2(N(C)C(c2ccc(NC(N)=O)cc2)=O)C1 CC1NC(=O)CCC1CNC(=O)C(N1CCC(Cc2nccs2)C1)=O c1(C(=O)NCC(CN(C(C(CC)C#N)=O)C)C)ncn2cc(Br)sc12 c1(CC(N2CCC(C)(NC(C=C(CC)C)=O)C2)=O)cccc2cnccc12 N1(C(C(C2CCCC(O)C2)(C)C)=O)CCC2(CCN(C(C3CCC3)=O)CC2)C1 C1(C(=O)NC2C(NC(c3csc(-c4ccccc4)n3)=O)C2)CC=CCO1 C(CCCCCN(C)C(c1cc(C(C)(F)F)n[nH]1)=O)NC(Cc1c(C)ocn1)=O CC1COCC(C(=O)NCc2cncc(CNC(C3(O)CCCCC3)=O)c2)O1 c1(N2CCC(CN(C(C3C(CC)CCC3)=O)C)CC2)cc(Cl)nc(C2(C)CC2)n1 c1(C(C(=O)NCCC(C)N(C(c2ccc(C)s2)=O)C)C)c(C)noc1C Cc1n[nH]c2cc(C(=O)NCC3CN(C(=O)CCN4CCCC4)C4CC34)ncc12 N1(C(=O)NCC)CCC(C)(C(=O)NOC(c2n(CC#C)ccc2)=O)C1 c1(C(N(C2CCC(NC(C34CC(C#N)(C3)C4)=O)C2)C)=O)ccc(F)c(O)c1 C1(N(C)C(=O)OC(C)(C)C)CC2CC1N(C(=O)NC1CCC(C(N)=O)CC1)C2 N1(C(C(=O)NC2(C)CCCO2)=O)CCn2ncc(S(C)(=O)=O)c2C1 C1(CC)CCCCC1C(N1CCCC1CC)C(=O)NC1CCOC1 c1(C(C)=O)ccc(-c2cn(C3CCC(C(N4CCCCCC4)=O)C3)nn2)cc1 C1(CC(=O)NC(COCCC)(C)C)CN(C(=O)C(COC)OCC)CC12CC2 C1(NC(c2c(C)nc(CC)s2)=O)CN(C(=O)CCCCC#N)C2CCCCC12 N1(C(CCC=CC)=O)CC2CCC1CC2NC(=O)CN1CCCCC1C CC1OC2(CNC(=O)CC3CCCCC34CC4)CC1(NC(c1csnn1)=O)C2 C(=O)(C(C(C)C)C(C)C)N1CCC(CN(C(CCc2cc(C)nn2C)=O)C)CC1 N1(C(CC)=O)CCCC(C(=O)NC2CCN(C(=O)COc3ccsn3)C2)C1 c1(C(=O)NCCC2(O)CN(C(C3(F)CCCOC3)=O)C2)cccnc1O c1(C(=O)OC)cc(Br)c(C)cc1NC(=O)C(=O)NC1CC(CSc2ccccc2)C1 C1(NC(C(C)NS(CCC)(=O)=O)=O)CN(C(C2(C#N)CC2)=O)CC(F)(F)C1 C1(CNC(C(C)OCC)=O)CCCC2(CN(C(=O)CCc3cncs3)C2)O1 C1(CNC(=O)C(O)C(F)F)CN(C(=O)C=C(Cl)Cl)CCC12CCOCC2 C1(C(=O)NCCCN(CCC)C(c2cc(C(F)(F)F)n[nH]2)=O)CN(CC)CCO1 C(CN=c1[nH]c2c(F)cccc2o1)=CC=CC=CC=C.CC1CCCCC1CC(=O)N c1(CNC(CN(C(=O)C2=C(C)CCC2)CCC)=O)cnn2c1CCCC2 S(=O)(=O)(c1cc(C(=O)NCC2CCN2C(C2(C)CC=CC2)=O)ccc1OC)NC Cc1cnc2c(C(=O)OCC=CC#N)c(C)nn2c1 Cc1nc2cc(C(=O)NCC(C3CCC(F)(F)CC3)C)cnc2[nH]1 N1(C(CC(CCC)O)=O)CCC2(CCC(NC(=O)C3=NOC(C)C3)CC2)C1 c1(NC(CCCOc2ccccc2)OC(=O)CN2CCN2)ccc2ccccc2c1 CC1CCOC(C(=O)N(C)CC=CC(=O)N(C2CC2)Cc2nc[nH]n2)C1 C1(NC(Cc2ccc(C)c(F)c2)=O)CC12CCN(C(C1CC=CC(O)C1)=O)CC2 CC(C(=O)NC1CC(CC(=O)Nc2cccc(C(F)(F)F)c2)C1)C(C)O c1(CN(C(C(COCC)n2cc(C3(C)CCCCC3)nn2)=O)C)ccc(F)cc1 Cc1ncccc1CC(=O)N(C)CC1CCCN1C(=O)C(C)c1cccs1 C1(NC(C(CC)CC)=O)CN(C(C2CCCS(=O)(=O)N2)=O)C2(CCOCC2)C1 C=CC1(CC(=O)NCC(C)(CC)OC)CN(C(c2cnc[nH]2)=O)C1 O=C(C1=NOC2(CCN(C(c3cncnc3)=O)C2)C1)Nc1cccc(I)c1Br n1(CC)nnc(C)c1C(=O)N(C)CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CCO1 Cc1noc(C)c1S(=O)(=O)NC1CC2CN(C(=O)CCCC(=O)C3CC3)CC2C1 C(=O)(C#CC1(CC)COC1)NCCOC1CCN(C(C(CC)C(=O)OC)=O)C1 c1(C(N(C)CC2(CNC(C3CNC(=O)N3C)=O)CC2)=O)csc(S(N)(=O)=O)c1 Cc1csc(C(N2CCC(OCCNC(=O)C(=O)N(C)C)CC2)=O)c1Cl Fc1ccc(Oc2ccccc2)c(CCCNC(c2c[nH]ccc2=O)C)c1 N1(C(C(F)OC)=O)CC2(C1)CN(C(c1c[nH]nc1Br)=O)CC2CO Cc1ccc(CCC(=O)NCCC2(CNC(=O)C(C)c3ccsn3)CC2)o1 C1(NC(=O)Cc2cncs2)COC2(CCCN(C(C3CCCC3)=O)C2)C1 c1(C(=O)NCCCOCCSCC(=O)Nc2n(C)cnn2)cccc(C=C=O)c1 N1(C(c2c(OCC)ccc(C)n2)=O)CCC2CC2(NC(=O)CS(N)(=O)=O)CC1 C1(CNC(c2scc(OC)c2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1(F)F C1(CC)(NC(=O)CC2(C)CC2(F)Cl)CCN(C(=O)Cc2cncs2)CC1 c1(OC)ccc(CCC(N2CCOC(C(C)NC(=O)COCCCF)C2)=O)cc1 c1(C(=O)NCCC(C(=O)N(CC(O)CO)C)OC)ccc(O)c(F)c1 C(C(C)C)(C(C(=O)NC)N(c1cccc(Cl)c1OC)C)OC c1(-c2scc(C(C)NC(=O)NC3CCC(C4CCNCC4)N3)n2)ccc(Cl)cc1 CCCCC(C(=O)N1CCC1C(C)O)NC(c1cccc(F)c1O)=O C(=O)(C(C)(O)CCC)N(C1CCN(C(C(C(=O)OCC)F)=O)CC1)C Cc1c(C(N2CCC(C)(NC(=O)CC(O)C(C)C)CC2)=O)sc2cncn12 C(C1CCCN1C(=O)CC1CCC1)=CC(=O)NCCCF c1(C(CNC(NCC)=NCc2cnn(C(C)C)c2)O)cccc(F)c1 CN1CCN(C(=O)CCc2cscn2)C(C(=O)NC2CN3CCCC2C3)C1 C(=O)(C(O)C(F)F)NCC1(C(C)NC(c2ncccn2)=O)CC1 Cn1cncc1C(=O)NCCCCCNC(C1(C2CC2)CC1)=O c1(OC)cncc(C=CCCNC(C2CCCC2(C)C)=O)c1 CC1(CNC(C2SC3C=CC2CC3)=O)CCN(C(C2CCOCC2)=O)CC1 Nc1c(F)ccc(Cl)c1C(=O)NC1CCN(C(=O)Cn2ncc(Br)n2)C1 CCCC(C(=O)NC(c1ccc(F)cc1)=O)OC(C1CCCN1CCC)=O c1(COC)cccnc1C(N1CCCC1CN(C)C(c1cn(C2CC2)nn1)=O)=O C1(C(=O)NCC(CC)(C)CC)CN(C(=O)Cc2ccc(C)c(C)c2)C(C)(C)C1 N1(C(C2CC(C)(O)C2)=O)CCN(C(=O)CCc2ccc(O)nn2)CC(O)C1 C1(CC=C)(NC(=O)Cc2cc(C)no2)CCN(C(C2CNC(=O)N2C)=O)CC1 c1(C(N2CCC(C)(C(N)=O)CC2)=O)ccc([N+](=O)[O-])cn1.c12ccc(c(F)c1)[nH]2 CC1=NOC(C(=O)NC(C2CN(C(=O)C3=CCCC3)C2)C)C1C c1(C(=O)O)cc2ncc(CN3CC4CC4C3CO)cc2[nH]1 C1(NC(CCC)=O)CCC2(CCN(C(C3(C)C=CCCC3)=O)C2)C1 c1(OC)nc(Br)ccc1S(=O)(=O)Nc1cnc2ccnn2c1 c1(-c2ccc(CN(C)Cc3c(OC)nsc3)cn2)ccc(Br)c(C)c1 C=CC1(CNC(=O)CC2CCCCN2C(C2CC(=O)NC2(C)C)=O)CCOCC1 C(=O)(C(C)(C)N(C)C)NCC1(N(C(CSCC=C)=O)C)CC1 C(=O)(C(C)CC(N)=O)NC1CCC(C(=O)Nc2c(C)oc(C3CC3)n2)C1 CC1CCOC1C(=O)NC1CC(CC=CC(N2CC(O)(c3cnn[nH]3)C2)=O)C1 c1(-c2cccc(OC)c2C)cccc2c(C(=O)NCc3ccc(CO)o3)n[nH]c12 C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(CSC(C)C)=O)C(CO)C1 C#Cc1cccc(CC(=O)N(C(CC)CC(=O)N(C(C)C(C)C)CC)CCC)c1 c1(OC)cc(CCN=C(NCCF)NC2CCCSC2)c(OC)cc1C c1(CC)ccc(C(=O)NC2(CF)CCC2)c(F)c1.c1(C(=O)N)n[nH]cc1 c1(C(N2CCC(N(C(CN(CCC#C)C)=O)CC)C2)=O)cccc2c1CCC2 N1(C(Cc2n(C)nnc2)=O)CCC(C)(C)CC1C(N1CC(CC(N)=O)C1)=O CC(C)(O)C(F)C(=O)NCC1(F)CC(NC(C2CC3CCC(C2)O3)=O)C1 C(=O)(C(C#N)C1CC1)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C C#Cc1cc(C(=O)NC(C)(CNC(c2cc(COC)on2)=O)CC)cc(F)c1 C1(C(=O)NCc2ccc(CC)cc2)CCCCN(C(C2CCCN(C)C2)=O)C1 N1(C(c2n[nH]c3c2CCC3)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1)CCO2 Cc1nc(-c2ncc[nH]2)sc1C(=O)NCCCC(C)(C)NC(=O)CNC=O c1(C(C(=O)NC(CC)CN(C(=O)CC(C)(F)F)C)N(C)C)ccc(F)c(F)c1 c1(OCC)ncccc1C(F)(F)F.C12CC3(C1)CC3CC(=O)N2 C1(CCNC(CCCOCCC)=O)CCCN(C(=O)CCC2CC(F)(F)C2)CC1 C1(NC(c2c(C)snc2)=O)CCC2(CC1)CN(C(c1ccc(CO)cc1)=O)C2 N1(C(c2cc(C(=O)OCC)on2)C(=O)NCCCSC)CC(C)OC(C)(C)C1C CC(C)CC(C)C(=O)N1CCC(N(C)C(c2cncc(OC(F)(F)F)c2)=O)C1 C[Si](C)(C)c1ccc(-c2csc(NC(=O)CCc3cccc(C(=O)O)c3)c2)cc1 C1(C(C)NC(=O)CN(C)C)CN(C(C2CCC(NS(C)(=O)=O)CC2)=O)CCO1 C1(O)(CN(C(c2c(C(C)C)ocn2)=O)C)CCN(C(=O)C=CC2(C)COC2)CC1 C(C(C)(C(=O)NCC1CCCN(C(c2ccc(OC(F)F)nc2)=O)C1)OC)OC C(CN=c1[nH]c(N2CCC(O)C(C)(C)C2)nc(=N)[nH]1)(C(C)(C)C)c1cn(CC)nn1 c1(C(=O)NCC2(F)CCN(C(=O)Cn3cc(CO)nn3)C2)cc2ccccn2c1 c1(OC)oc(C)nc1C(=O)NC1CCCC1NC(c1cc(C2CC2)ns1)=O c1(OC)cc(C)c(C(c2nnnn2C2CCC2)NCc2conc2C(C)C)cn1 N1(C(CC(COC)C)=O)CC2(C(=O)NC(CCO)C3CCCC3)CC1CCO2 C(=O)(C1CCOc2ccccc21)NCC1(C)CC(NC(c2cc(C)c(C)s2)=O)C1 c1(OC)cncn(CC(C)NC(c2cccc(Br)c2)=O)c1=O C(=O)(CC(O)(C(F)(F)F)c1ncc[nH]1)N1C(CNC(=O)CC2SCCS2)CC1 Cc1ccc2c(C(=O)NC(CNC(=O)C(C3CCOCC3)O)C3CC3)n[nH]c2c1 N(C1CCCc2c[nH]nc21)C(C(N1CCC(CC#C)C1)=O)=O C1(C)(NC(c2ccc(C(C)C)cc2)=O)CCCN(C(=O)C2=COCCC2)C1 Cn1nc2ccccc2c1Cn1cc(-c2ccc(Cl)c(N)c2)nn1 CCC(C)(C)C(CC(=O)N1CC(c2ccccc2C(F)(F)F)C1)NC(C)=O C(CC(=O)NCCC(=O)NCCC1(C(=O)NC)CC1)SCCC c1(CN2C(C(N(C)CC#N)=O)CSCC2)cc(Cl)cnc1Br C1(C)(C(c2n(CCCCCC)nnn2)NCc2cc(C(F)F)no2)CC=CCO1 CCC(CC(=O)N1CC(O)CC1c1ccc(F)cc1)C(C)(C)C C1(C(=O)OC)CCC(C)(C)N(C(=O)CCc2cn(C(C)CO)nn2)C1 O=C(C1=CCCN(C(C23CCCN(CC2)C3)=O)C1)NCC1CSC1 N1(C(c2c[nH]c3cccnc23)=O)CCc2c(F)cc(F)cc21 Cc1ncc(C(=O)NC23CC(CNC(=O)CC4CC4C)(C2)C3)cn1 c1(C(N(CCNC(=O)C=CBr)C2CC2)=O)ccc(C2CCOCC2)cc1 CN1CCC(CN(C(=O)C(CC2CCCC2)NC(=O)CCC2CC2(C)C)C)C1 c1(C(=O)NC(CNC(C2C(=C)CC2)=O)(C)Cn2cccn2)ccc(F)nc1F C(=O)(C1=NN(c2ccc(C)cc2C)C(=O)C1)NCC1C2CN(C(CC)=O)C1C2 c1(CNC(c2occ(C)c2)c2nnnn2C)cccc(C(F)F)c1 N1(CCC)CCN(C(=O)CCC2CCCN(C(C3CCCS3)=O)C2)CC1 c1(C(=O)NC(CN(C(C(C)=CC)=O)CC)C)c[nH]c2cc([N+](=O)[O-])ccc12 c1(C(C)C)ccc2c(c1)CN(C(=O)NC1CCN(C(c3ccccc3)C)C1)C2 C(=O)(C(CC(C)(C)C)NC(C1C=CCN(C(C2CCCCN2C)=O)C1)=O)OC c1(CN(S(C)(=O)=O)C)cn(C(C)C(=O)NC2CC(CO)C2)nn1 c1(N2CCC(C(C)NC(c3csc(-c4ccco4)n3)=O)C2)ncn(C)c(=O)c1Br N1(C(c2ccc(CC)nc2)=O)CC(C(=O)NCC=CBr)C(C)(C)C1 C1(NC(C(C)C2CC2)=O)CCN(C(=O)Cc2ccco2)C12CC2 N1(C(c2cnc(O)c(F)c2)=O)CC(NC(C2CC(F)C2)=O)CC2(CC2)C1 C(=O)(CS(=O)CCC(F)(F)F)NC1(C2CCN(C(c3ccn(CC)n3)=O)C2)CC1 N1(C(c2c(SC)nn(C)c2)=O)C(CNC(C2CC2[N+](=O)[O-])=O)CC2CCCC12 N1(C(c2c(C)ccs2)=O)CC(=O)CC1C(=O)NCC1CCCOCC1 C#CCCCCCC(=O)N1CCCCC1C(C)NC(c1c(C)ncn(C)c1=O)=O C(=O)(C(F)(F)C(O)C(C)C)NC1C=CCN(C(c2ccc(S(=O)(=O)NC)o2)=O)C1 Cc1c[nH]nc1C(N1CCC1CC(=O)NCC1(N(C)C)CCSC1)=O CCC(CC1CCCC1)C(=O)NCCOCCCNC(C1CSC(C)=N1)=O c1(C(N2CC(C(C)C)OCCC2)=O)ccc2ncccc2c1 c1(OC)cccc(C(C)(C)C(=O)N2CCC(NC(c3cnc(CSC)s3)=O)C2)c1 c1(C(=O)OC)ccc(CC)c(NC(=O)NN2CCOC3(CCSC3)C2)c1Cl CC1(O)CCC(CC(N2CCC(O)(CNC(c3cc4n(n3)CCO4)=O)C2)=O)CC1 c1(C(=O)NCC2CCN(CCn3cccn3)C2)cnc2c(c1)CCCO2 C1(C(=O)N(C2C(=C)CC2)CC)CC1C1CCN(C(=O)Cc2cc(F)cc(F)c2)CC1 N1(C(CCc2c(C)noc2)=O)CCCCC(C(=O)NCCCCN=[N+]=[N-])C1 Cn1ncc2nc(Cl)nc(NC(CNC(c3ccc4nc[nH]c4c3F)=O)CO)c12 N1(C(C2(CC=C)CC=CC2)=O)CCCCC(C(N2CCCC(N(C)CC)C2)=O)C1 C(=O)(C1=COCCC1)N1C(CN(C(=O)C=Cc2cscn2)C)COCC1 C(=O)(C(C(C)NC(=O)Cn1cc(CN2CC3CCC2C3)nn1)C(C)C)NC N1(C(c2cc(C)c(Cl)cc2)=O)CCCC2CN(C(=O)C#CC3CC3)CC12 c1(NC)ccc(C(N2CC(NC(=O)CC(C)C(C)C)CCC2C)=O)c(Cl)c1 C1(CC(N2CCC(CNC(=O)CC(F)F)C2)=O)CCCOC1 N1(C(CC=C)=O)C(C(=O)NCCn2cc(COC)nn2)CC1C N1(C(C(C(CC)CC)C)=O)CCCCC12CC(NC(C1CCCC1)=O)C2 c1(C(=O)NC(CC)CNC(=O)CCc2ccc(OC)cc2)ncc2n1CCCC2 CC1(C(=O)OCc2cccc(-n3ccnc3)n2)COC(C)(C)OC1 N1(C(CCCOCC)=O)CCOC2(CCCN(C(=O)C3=C(CC)OCCS3)C2)C1 C=C1CC2(C1)CC(C(N1CC(N(C)C(c3cc(Cl)cc(Cl)c3)=O)C3(CC3)C1)=O)C2 C#Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)Cc2ccc(Cl)cc2C)cc(F)c1 C1(CNC(c2c(C)noc2C2CC2)=O)CN(C(C2CC(=O)N(C)C2)=O)CC1(F)F C1(C)(C(N2CCCC(N(C(CCOCCOC)=O)C)C2)=O)CCCCC1(F)F c1(CC(N2C(CNC(=O)CCC3CCOC3)C=CC2)=O)ccc2c[nH]nc2c1 C1(C(N(CCCNC(c2cnn[nH]2)=O)C)=O)CCCCO1 N1(C(C(CN(C(CCC(C)(C)OC)=O)C)C)=O)CCOC2(CCC2)CC1 N1(C(=O)CCOc2ccc3ncccc3c2)CCCc2c(F)ccc(Br)c21 Cc1ccc(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C2)c([N+](=O)[O-])c1 c1(OC(C2N(C)C(NC(=O)OC(C)(C)C)CC2)=O)cc2oc(O)nc2cc1F C(N=c1[nH]c2c(c(=NC3CC(C(N)=O)C3)[nH]1)SCC2)c1nc(CC)sc1 N1(C(C(C)CN(C(=O)CC2CCC(=O)N2C)C)=O)CCC12CCCC2 c1(C(=O)O)cnc2n1CCN(C(c1ccn(-c3ccccc3)c1C)=O)C2 N1(C(C(C)OC(=O)OCC)=O)CCC2(CC2NC(c2cccnc2C2CC2)=O)C1 c1(C(N(C2CC(O)CC(C)(C)C2)c2c(C)n(C)cn2)=O)ncc([N+](=O)[O-])n1C Cc1cc(C(N2CC(O)(Cc3cn(CCF)nn3)C2)=O)c(N)c(F)c1Cl c1(CN2CC(CC)N(C(=O)Cc3cnc(OC)cn3)CC2)cc(Cl)c(C)cc1O N1(C(C=Cc2c(OC)cccc2)C(=O)NC(C)C)CCOC2(CCCSC2)C1 c1(C(=O)NC2C(NC(C(C(=O)OC)(C)F)=O)CC2)nccc2ncccc12 N1(C(c2cc(C(C)(C)C)no2)=O)CCC(O)(CNC(C2C=CCS2)=O)C1 c1(CC(C)C(=O)NCC(F)CNC(=O)C2=CCSC2)ccccc1Br c1(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CC2)cc(O)c(O)c(O)c1 c1(C(=O)NC(CC)CNC(=O)CSc2cn[nH]c2)ccc2nc(O)oc2c1 C1(CNC(c2n[nH]c(CC)c2Cl)=O)CCN(C(C2CCCC2(C)C)=O)C12CC2 Cc1coc(C)c1C=CC(=O)NC1CC1NC(=O)Cn1cnc([N+](=O)[O-])c1 C1(NC(c2c(C)[nH][nH]c2=N)=O)CCCN(C(c2ccc[nH]2)=O)CC1F C(CCCC(=O)N(C)CCO)NC(C)=O.c1(CCN(CC(=O)NC)C)ncc(F)cn1 Cc1coc(C(N2CCCC2CCNC(=O)CCc2c(C)noc2Cl)=O)c1C c1(C(N2CCC3(C(N(C(C)C)C)C3)C2)=O)cc2cc(F)ccc2s1 N1(C(c2ccn(CCC)n2)=O)CC(C(=O)NC2(C(C)C)CCC2)C2(CCC2)C1 C(=O)(CS(=O)(=O)CC(C)C)NCC1N(C(C2C(OCC)C2C)=O)CCC1C N1(C(c2nnsc2C(F)F)=O)CC2CC(C1)N(C(C1CCc3nnnn3C1)=O)C2 CN=c1nc(C(=O)NC2CC(CNC(=O)C(C)(C)CC)C23CCC3)cc(C)[nH]1 N1(C(CC(CC2CC2)NC(c2c(C)c(O)ccc2)=O)=O)CCC(F)(F)C(O)C1 c1(CCC(=O)O)ccc(CNC2CCCCC2n2ccnc2)nc1 C1(CCNC(C2CCCC2O)=O)CC2CCC(C1)N2C(c1cc(CCO)on1)=O c1(SC)cc(C)ccc1C(N1CCCC(CNC(=O)CN2CC(C)(C)C2)CC1)=O c1(C(N(CCN(C(c2ccc(CC)s2)=O)C)C)=O)[nH]ncc1C#N N1(C(COCCCOC)=O)CC(C(N2CC3CC2CC3C)=O)CC(C)C1 N1(C(C(CN(C)C)(C)C)=O)CC(=O)NCC1C(N)=O C1(C(=O)NC(C=C)CO)CCC(C)N1C(=O)CCc1ccc(OC(F)F)cc1 C(CC1=CCN(C(C2CCN(C)C(=O)C2)=O)CC1)NC(c1c(Cl)cc(C)s1)=O N1(C(c2c(CNC(C)=O)nccc2)=O)CCC(F)(NC(=O)COCC(F)(F)F)CC1 c1(C(N2CC(CN(C)Cc3nnc(C)o3)OCC2)=O)cc(C)c(C#N)c(C)c1 C(C)(CCC(=O)NC1(CO)CC=CC1)NC(C(C)n1cnnn1)=O C1(CCC(=O)N(CC#C)CC2CC2)CCCN1C(=O)C(C)[SH](CC(C)C)CC C1(CN(C(C=CCC)=O)C)CCCN(C(=O)C=Cc2cncn2C)C1 N1(C(CONC(=O)CCc2ccco2)=O)CCC2(CCCOC2)C1.C1(N)(CO)CCC1 N1(C(c2cccc(C)n2)=O)CCC2(CC1)CCN2C(C1C=CCN1)=O Cc1cnn(C)c1S(=O)(=O)NC(=O)CC(C(N)=O)C1CCC1 C1(NCc2c(C)cc(C(=O)O)nc2)CCc2n[nH]cc2C1C N1(C(C2C=C(C)CS2)=O)CC2OCC(NC(c3cccc(F)c3)=O)C2C1 CC1C(C(=O)N2CCC3(CCCN3C(=O)C#CC3(C)CC3)C2)=Cc2ccccc21 N1(C(CC(C=C)CC)=O)CCCC2(CCN(C(=O)CC(C)(C)C)CC2)C1 CC(=O)CC(C)(C)CC(=O)NCC1CC(NC(c2cnoc2)=O)C1 c1(C(=O)NCC2CCCC(NC(C(C)=C3CC3)=O)C2)oc2ccc(Cl)cc2c1C N1(C(=O)O)CC2CC(C1)N2C(C1CCCCC1CN)=O.CC(C)(C)C(=O)CC1CCC1 O=C(CC(F)(F)Cl)NCC(CO)NC(c1ccc(-c2nc[nH]n2)nc1)=O c1(C(=O)NCC2(C)N(C(C(C=C)O)=O)CCC2)ncn2cccnc12 CC(C)(CCC#N)C(=O)NC1CC1NC(c1ccc(C2CCOC2)s1)=O c1(C(=O)NC(CC)CN(C)C(C2(OC)CCC2)=O)cnc(OC)c(Cl)c1 CON(C)C1CN(C(c2nc(CNC(=O)Cc3ccccn3)oc2C)=O)C1 C1(NC(CCNC(C2C(C)C2)=O)=O)CCC(CNC(=O)C(C)(C)c2nncn2C)C1 C1(NC(c2c(CC)n(C)nc2)=O)CN(C(c2cccc(N)c2F)=O)CC(C)(C)C1 c1(C(=O)NCC2C(CNC(c3cn(CCC)nn3)=O)C2)ccc(O)c(C(N)=O)c1 N1(C(C=CC(C)(C)NC(C2CC23CCOCC3)=O)=O)CCC2(CCCCO2)C1 CC(C)CC(C)CC(=O)NC1(C)CC(C(=O)NC2CC3CCCC3C2)C1 Cc1ccc(COC(=O)C=CCC(=O)C(C#N)c2nccs2)c(Cl)c1 C1(COC)CCN(C(C2CC(NC(C3(C)CC3)=O)C2)=O)C1(C)C C1(CC)CN(C(=O)C2CC2)CC1C(=O)Nc1csc(Cl)c1 CCCC(C(=O)NCc1c[nH]nc1C(=O)NC1CNC(=O)C1)OCC C1(CNC(c2n(CC)ncn2)=O)CCN(C(=O)C(N2C(=O)CCC2=O)C)CC1 N1(C(C(C2CC2)OC)=O)CCCCC2(CCN(C(=O)CNC(=O)CCCCO)C2)C1 C#CCCCCCC(=O)NCCC1CC(C(=O)NCC2CCN(C(C)=O)C2)C1 C1(NC(c2ccsn2)=O)CN(C(=O)C=CC(c2ccccc2)=O)C2(CCC2)C1 n1(C(CC)(C)C)nnc(CO)n1.n12nnnc1C(NCCc1ccc(C)o1)C2C Cc1cc(C(N2CCC(C)(C)C2CNC(=O)C(C2CC2)C2CC2)=O)cc(C)c1F c1(OC)ccn2cc(C(=O)N(CCNC(c3csc(C)c3)=O)C(C)C)nc2c1 c1(C(=O)NC2CN(C(c3c(CC)cco3)=O)C2)ccc(C(C)(C)NC(C)=O)cc1 CC1(C#N)CCC(CO)(NS(=O)(=O)CC2CCCNC2=O)C1 c1(NC(=O)NCc2nccc(OC)n2)cc(C)ccc1Br N1(C(CC2CCCC(C)O2)=O)CC2(CCN(C(=O)CN(S(C)(=O)=O)C)CC2)C1 C(=O)(C(C(C)C)NC(c1ncc(F)cn1)=O)NC(C(=O)NCC(C)C)C C=CCC(C)(CC=C)NC(=O)C1=NOC(CNC(=O)CCc2csnn2)C1 CC(C)C(O)C(F)(F)C(=O)NC1CN(C(=O)C=Cc2ccc(Cl)cc2)C2CC12 N1(C(C(CC)OCC2CC2)=O)CCOC(C(=O)NOCC(O)C(C)C)C1 c1(C(=O)NCC(=O)NCC(=O)NC(C(C)C)C(=O)N(C)C)cnn2c1N(C)CC2 c1(CNC(=NC)NCC2CC(C)=NO2)ccc(N2CCOCC2)cc1Cl C=CCCCC(=O)N1CCC1(C)CC(N1CCCC1C1CCOC1)=O C1(C(N(CC#CC)CC#C)=O)CCCCCCN1C(=O)C(C)OCC=C N1(C(c2cnc(C(C)C)o2)=O)CCCCC(C(=O)NCC2OC(=O)CC2(C)C)C1 c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)ccc(N2CCCCCC2)cc1 C(=O)(C(C(=O)N1CC(OCC(=O)NC2(C)CCN(C)CC2)C1)C(C)C)OCC C(CCC(C(=O)NC1C2CCCC12)NC(=O)C(C)CC#N)OC c1(C(N2C(c3cn(CC(C)O)nn3)CCCC2)=O)ccn(CC(F)F)c(=O)c1 c1(C(=O)NCC(CCCC)NC(c2cocc2C)=O)cnc2c(cnn2C)c1 c1(-c2ncc(C)s2)nc(C2CCC2)nn1C1CCCCC1 CCCCCC(=O)NCC1CN(C(=O)Cn2cnc(C(F)(F)F)n2)CC1O c1(C(N(CC(C)(C)NC(=O)Cc2nccn2C)C)=O)c(F)ccc2c1OCC2 C#CCC(C)(CC)C(=O)N1CC2CCC1CC2NC(=O)C(C)NC(=O)CC O(NC(=O)C(CNC(=O)C1=NOCC1)CC1CC1)CC c1(NC(C(CC2CN(C(C3=NOC(C)C3)=O)C2)F)=O)ccc2ccncc2c1 c1(C(C(N2CCN(C(=O)CCOC(=O)N(C)C)CC2)C)=O)cc(Cl)sc1Cl N1(CC)CCCC(N=c2[nH]c(=NCC3(CC4CC4)CCC3)[nH]c3c2CSC3)CC1 CC1=C(C(=O)NC(c2cn3ccsc3n2)=O)CCC1.C12CN(CCC1C)N2C c1(OC(N2CCC(OCC(=O)OC)C2)=O)cc(OC(C)(C)C)cc(Cl)c1 C1(N(C(=O)CCn2cnnn2)C)CCC(NC(c2cnc(S)[nH]2)=O)C1 C(C)(C(=O)N1CC(O)CO1)N(CCCCCNC(C)=O)C N1(C(C)=O)CCCC(NC(=O)CCN(C(=O)C=Cc2cc[nH]n2)C)C1 c1(CC(=O)NC(C2N(C(c3nc(SC)sc3)=O)CCC2)(C)C)cncc(C)c1 N1(C2(C(=O)NC3C(NC(c4cn(CCOC)nc4)=O)CC3)CC2)C(=O)CCC1=O O=C(CCCCC(F)(F)F)NC1CN(C(c2ccc3c(c2)CCO3)=O)CC2CC12 N1(C(=O)NC2CCCC(C(N)=O)C2)CC2CCC1C(O)C2O Cc1nc2ccc3cc(C(=O)NC4CCN(CCC5CCOC5)C4)ccc3n2n1 c1(CC)cc(F)ccc1CC(=O)N(C1CCCN(C(C2(Cl)CC2(C)C)=O)C1)C c1(NC(C2(CC#C)CCCO2)=O)cccn(-c2ccccc2)c1=O Cc1nc(C(=O)NC(C)CCCNC(C2(C)CC=CCC2)=O)cc(O)n1 c1(C(=O)NC(C2CCN(C(=O)C(Cl)=CCl)C2)(C)C)cnc2ncccc2c1 CCCCC(C(=O)NC1CCN(C(c2ccc(CC)nc2)=O)C1)ON=C(C)C N(C(=NCc1ccc(Nc2ccncc2)cc1)NCC1CCC1)C1C(C)(C)C1 C1(C(N2CCC2C(=O)OCC)=O)(CNC(C2N(CC)CSC2)=O)CC12CCC2 c1(NC2CCC(CC)CC2)cc(NCCS(=O)(=O)NC(C)(C)C)nc(C)n1 Cn1cc(C(N2CC3CC3(CNC(C3(C(F)F)CCCO3)=O)C2)=O)c(C(N)=O)n1 N#Cc1cccc(CC(=O)NCC23CC(NC(=O)Cn4cnnn4)(CO2)C3)c1 c1(C(=O)NC(C2N(Cc3c(CC)cccc3)CC(O)C2)=O)ccc(CO)c(F)c1 N1(C(c2c(CC)cccc2)=O)CC(NC(c2occc2F)=O)CC(F)(F)C1 c1(C(=O)NC2C(NC(=O)COC3CC3)CC(F)(F)C2)cc(Br)cnc1O C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(SC)C(NC(=O)COC(C)(C)C)C1 c1(SCC)ccc(C(=O)NC2CCOC2)cc1.c12cn(nn1)CC1CN(C1)C2=O c1(CC(=O)NCC2CCN(C(=O)CCCC3CC3)C2)csc2cccc(Cl)c12 c1(C(N2CC(C(O)C(F)F)C2)=O)cc(F)ccc1OC(F)F CC1(C)CCOC(C(=O)NCC#CC(=O)NC(c2ccccc2)(C)C)C1 C1(C(=O)NCCC2CCN(C(=O)Cn3cnc(Br)c3)C2)CCCS(=O)(=O)C1 c1(C(=O)NCC2(NC(C=CCC)=O)CC2)cccn2ncnc12 c1(CC)ccccc1C(=O)NC1CCCC(NC(=O)CCCNC(=O)C2CC2)C1 c1(SC)nc(N2CC(C(N)=O)(CNC(C3CCCCC3C)=O)C2)ncc1C C#Cc1ccc(F)c(C(=O)NC(C2CCCC2)CNC(C2(Cl)CC2(C)C)=O)c1 c1(C(N2CC(NC(C)=O)CC(OCc3ccccc3)C2)=O)cc(F)c(F)cc1O C1(CNC(c2ccn(CC)n2)=O)CC2COCC2N1C(=O)CCN1CCCCC1 C1(C(=O)NC2CN(C3(O)C(CC(=O)N(CC)CC)C3)C2)CC(OC)(OC)C1 CC1C(NC(=O)Cc2cc(Cl)ccc2Cl)CCCN1C(=O)Cn1cccnc1=O Cc1ccc2c(c1)CCC2Nc1conc1C1CCCC1 C1(CNC(C(C(COC)C)C)=O)C(C2CC2)CCN1C(=O)C(CCOC)OC C(=O)(N=c1ccc(Cl)n[nH]1)C1(C)CCN1C(c1csnc1-c1ccccc1)=O C1(NC(C2CC3CC3C2)=O)CCN(C(c2ccc(COC(F)(F)F)cn2)=O)C1C C(C(=O)NC1CC(CCNC(=O)C=Cc2ccccc2)C1)(C(C)C)OCC CCS(=O)(=O)C=CC(=O)N1CC(C(C)NC(c2cc(OC)ncn2)=O)C1 c1(C(=O)NC2CCC(NC(c3cnn(-c4ccccc4)n3)=O)C2)ccc(F)cc1 N1(C(CC2(C)N(C(C(C(C)C)C3CCC3)=O)CC2)=O)CCCC(O)(C2CC2)C1 c1(OCC)cc(C(C(=O)NC(C)C)N(CCCN(C)CC#N)C)ccc1C c1(C(N2CCCC2Cn2cc(CCC#N)nn2)C)ccoc1-c1ccccc1 CC(N=c1[nH]c2c(c(=NCCC3CC(C)(C)NC3=O)[nH]1)CCC2)C(C)F S(=O)(=O)(c1ccnc(NC(c2ccc3c(c2)CN(C)C3)=O)c1)N(C)C N1(C(C(N)C2(n3cc(-c4ccccc4)nn3)CC2)=O)CC2C(C(=O)NCCl)C2C1 C1(C(=O)NCC(CNC(CCc2onc(C(C)OC)n2)=O)(C)C)CCCOC1C C1(NC(C(CC)O)=O)(CC)CCCN(C(c2cnn(C3CCOCC3)c2)=O)C1 N1(C(C2OCCN(C(c3cccc(OC)c3)=O)CC2)=O)CCC(O)C12CCCC2 C(C(C)C(=O)N1CC2CC2C1)N(C(COC(CC)(C)C)=O)C N1(C(c2cccc(C)n2)=O)CCN(C(c2sc(C)cc2Cl)=O)C2CCCCC2C1 N1(C(C=CC(=O)OCC)=O)CCC(C)(CN(C(C2CC(C(C)C)C2)=O)CC)C1 c1(SC)nc(C)c(CC(=O)N(C)C(c2cn(C3C4CCCCC34)nn2)C)s1 c1(C(N2CCN(C(c3scc(C)n3)=O)CC2C(F)(F)F)=O)cc(I)c(O)cc1O c1(NC(c2ccc(Cl)cc2)C(=O)NCCC2(C)CC2)cccnc1Cl N1(C(C2CCN(C)CC2)=O)CCCCC2(CCN(C(C3CC4CC34)=O)C2)C1 c1(CN(c2nccc(NCCCC)n2)C)c(Cl)cccc1Cl C(=O)(CCN=c1ccc(C)c[nH]1)N1CCN(C(C(CC)(CC)CC)=O)CC1 CCC(C)CC(=O)NC(CC)C(=O)N(C1CCNC1=O)C c1(CC)ccc(C=CC(=O)N(C2CC(NC(C3C(C)C3(F)F)=O)C2)C)cc1 C(C1CCCCC1)=CC(=O)NC1(C(=O)NCC(COC)OC)CC(CO)C1 N1(C(c2c(OC)c(C)sc2)=O)CC2CC(NC(c3c(C)nn(C)c3Cl)=O)CC1C2 C1(COC)(NC(=O)CC(C)O)CCN(C(=O)CCSc2ccccc2)CC1 C=CC(C)CC(=O)NC(C(=O)NCCC(C)(C)F)C1CC1 c1(C(=O)NCC2N(C(C3(C(=O)OC)CCCO3)=O)CCOC2)cc(C)cc(Cl)n1 N1(C(C(C)(CO)NC(=O)CCC2CCOC2)=O)CCNC(=O)CC1 N1(C(Cn2c(C)c(Br)cn2)=O)CC(C)(C)CC1CNC(=O)C(C)CF c1(C(N(CC(C)NC(C2CC2c2ccc(Cl)s2)=O)CC)=O)csc2cncn12 CC1(C(=O)NC2CC(NC(=O)CC3(c4ccccc4)CC3)C2)CCCO1 N1(C(C2C(C)=CCC=C2)=O)CCN(C(c2ccccc2)=O)C(CC#N)C1 C1(NC(=O)COCCOCCO)COCCN(C(=O)C2=C(Cl)CC2)C1 c1(C(C)C)ccsc1C(N1CCC(c2cn(CCNS(C)(=O)=O)nn2)C1)=O C12(CNCCOc3c(OC)cccc3)CC3CC(CC(C3)C1N)C2 C12(NC(C3CN(C)C(=O)C3)=O)CCC(NCc3ccc(CC(=O)O)cc3)(CC1)C2 N1(CC)CCN(C(=O)C(C)N(C(c2cn3c(n2)CCC3)=O)CC)CC1C N1(C(C2CCc3nc[nH]c3C2)=O)CCOC2(CCCN(C(=O)C(Cl)(Cl)Cl)C2)C1 c1(N2C3CN(C(c4c(S(C)(=O)=O)ccs4)=O)C(C3)C2)ncnc2sc(F)cc12 c1(CN(c2ccc(C#N)nc2)C)cccc2c1S(=O)(=O)CCC2 N1(C(c2cc(C(=O)OC)oc2)=O)CCC2(CC1)CN(C(=O)C=CCO)CC(C)O2 Cc1cccnc1CNC(=O)CN(C(c1c[nH]c(C)c1)=O)CC1CC1 CC(CC(F)(F)F)C(=O)N(CCCN(C)C(C1CC2(CCCC2)CO1)=O)C CC1CCCC=C1C(=O)N(CCCNC(=O)CCc1ncc(F)cn1)CCO CS(=O)(=O)c1cncc(-c2ccc(C(=O)N(CC(F)(F)F)CC#N)nc2C)c1 c1(OC)ccc(C)c(C(=O)NCCC23CCC(C2)N(C(=O)CNC(C)=O)C3)c1 c1(C(N(CC(CC)NC(C(CCC)OC)=O)CC)=O)cc2cc(C)ccc2o1 C1(C(=O)NC2(C(O)CO)CC2)CC(O)CCN1C(C1CCC2CC1CO2)=O Nc1ccc(-n2cc(CONC(C3CSCCN3CC(F)(F)F)=O)nn2)cc1 C1(N(C)C(c2cncs2)=O)CC2CC1N(C(=O)C(c1ccccc1F)(C)F)C2 CC(C)(C(=O)NC1CCC(CNC(C2CC3CC3C2)=O)C1)c1cccs1 N1(C(COC(C(=C)C)=O)=O)CC2(CCN(Cc3cc(Cl)ccn3)CC2)C1 c1(C(N2CCCCC(CCC(N3C(C#C)CC3)=O)C2)=O)cccc2ccoc12 N1(CC)CCCN(C(C2CC3CC3N2C(c2ccc([N+](=O)[O-])o2)=O)=O)CC1 N1(C(c2cnc[nH]2)=O)CCC(C(CO)NC(C2CC=CCC2)=O)CC1 c1(OC(C(=O)NC(CCCNC(C(COC)(C)C)=O)C)C)cc(C)ccc1Cl C1(C(=O)NCCN(C(c2ccc(N)cn2)=O)C2CC2)CCN(CCO)C(=O)C1 CN=c1nc(C(=O)NC2CN(C(C3CCCN3C=O)=O)CC2C)cc(C)[nH]1 N1(C(c2c(Cl)ccc(OC)n2)=O)CCCCCC(NC(=O)C(C)(C)CF)C1 C1(C2(NC(c3cc(Cl)c[nH]3)=O)CC2)CCCCN1C(=O)C=CC1CCOC1 C1(NC(c2c(C(C)C)n(C)nc2)=O)CCC2(CCN(C(C3SCCCS3)=O)C2)C1 c1(OC)cccc2c(N3CCOC(CNC(=O)CCn4cncn4)C3)ncnc12 N1(C(Cc2n(C)cnn2)=O)CCCCC(NC(=O)CCn2ncn(C)c2=O)C1 Cc1cc(Br)oc1C(=O)NC1CC(C)N(C(c2ccsc2Cl)=O)C1 CC(N=c1[nH]c(=NCC2CCSC2)c2c(F)cccc2[nH]1)c1cc(Br)ccc1Cl N1(C(c2c(CC)ncs2)=O)Cc2n[nH]cc2C1C(=O)N1CCC(C(=O)NC2CC2)C1 C(C(C)(C)C(=O)NCCC(C)N(C(=O)Cn1cncn1)C)OCC CC1(C)CN(C(c2cnc[nH]2)=O)CCN(C(c2ncoc2Br)=O)C1 c1(C(N2C(CNC(CC(C)F)=O)CC(O)C2)=O)ccc2cccnc2n1 c1(NC(CC2(OC)CN(C(C3CCCN3C(N)=O)=O)C2)=O)ccc(F)cc1O c1(C(N2CCC(CN(C(CC=CCC)=O)C)C2)=O)ccc(C(F)(F)Br)nc1 C(CCN=C(NCC1CC2(CCOCC2)O1)N1CCCC(CC(C)(C)C)C1)OC N1(C(C2CCN2C(C2CCCC2F)=O)=O)CCc2ncccc2C1 C1(NC(c2c(C#C)c[nH]n2)=O)CCCCN(C(=O)CCCn2nc(C)cc2C)C1 Cn1cc(C(=O)NCC(C2CCN(C(C3C=CCCC3)=O)CC2)F)c(O)n1 N1(Cc2c(OC)ccc(F)c2)CC2C(C1C(=O)NC1CC(O)C1)C2(C)C C1(C(=O)NC2CC(OCC3CC3)C2)CCN2CCCC2C1 c1(CNC(c2c(C)occ2)=O)cccc(C(N2CC[Si](C)(C)C2)=O)c1 c1(CCC(=O)NCCC(C)N(C(=O)C2=NNC(=O)CC2)C)ccc(C#N)cc1F CC1CCC(Cl)=C(C(=O)N2CCCC2CNC(c2cc(Cl)cn2C)=O)C1 CCC(C(=O)OC)C(=O)NCC1CCCCN1C(c1cc(Cl)ccc1F)=O CC1C(NC(c2ccnc(F)c2)=O)CC2CCC1N2C(C1CCCN1C=O)=O N12CC3C(CS(=O)(=O)C3C1)C2=O.CC1CC(C)(CNC(C)(C)C)C1 c1(C(C)NC(C(=O)N(C)Cc2nnc(C(=O)OCC)s2)=O)ccc(C)cc1F c1(CC(=O)NCC(C)CNC(C2(C3CC3)CCOCC2)=O)cccc2sccc12 Cc1noc(C)c1C(C(=O)NC1COC1)N(c1ccccc1)C1CC1 Cc1ccsc1CNCC1(c2ncccn2)CCOC1 C#Cc1ccc(C(=O)NCc2occc2C(=O)NCC2CCOCC2)o1 c1(CNC(c2c(CC)[nH]cc2)=O)ccc(C(C)NC(=O)C(C)(C)OC)cc1 c1(C(N2C(C)CC(CC(=O)NCC(C=C)(C)C)C2)=O)c(C)nn(C)c1N C1(C(=O)NC(C)CC2CCC2)COC(CNC(=O)C(Cl)Cl)C1 c1(CC(=O)NCC2CCCCN(C(CSCC#C)=O)C2)ccc2c(c1)CCCC2 N1(c2nnc(C3C(CC)CCO3)n2CC2CC2)CCOC2(CCCC2)C1 c1(C(N(C2CCN(C(c3cccc(NC(C)=O)c3)=O)C2)C)=O)nc(C)ccc1C c1(C(=O)NC2C(NC(C3CN(C)C(=O)N3)=O)CC2)cc(Cl)ccc1F C(CCN=C(NC1CC(C)(C)C1)NC1CCCCC1C)OC(C)C N1(C(C2CCC(C)(CC)O2)=O)CC2(CC(CNC(c3cnc(C)[nH]3)=O)C2)C1 Cn1c(C(N2CCCCC2CCNC(C2CC(=O)NC2(C)C)=O)=O)cccc1=O C1(NC(C2C(C)CC(=O)N2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 C1(C(=O)NC2CCC(NC(C(C)N3CCC3)=O)CC2)Cc2nncn2C1 Cc1cccn2ncc(C(N3CCC4C(CCN4C(=O)COC4CCC4)C3)=O)c12 c1(C(=O)NC(C2(O)CN(C(C3COC3)=O)C2)C)cc(C(C)(F)F)ccc1C C(=O)(C(Cc1cnc[nH]1)NCC(=O)NC(C)(C)C)NCC=C(C)C C1(c2cn(C3c4ccc(o4)C(=O)N4CC3C4)nn2)(CC)CCOC1.OC.OC C(=O)(CCCCCOC)N1CCC(C(CNC(C(CC)OCC2CC2)=O)C)CC1 N1(C(Cn2nnc(C)n2)=O)CC2CC1CN(C(=O)CCSc1ccc(F)cc1)C2 C(=O)(C(C)(C)C(F)F)NC1C(CNC(c2cc(OC)no2)=O)CCC1 C(CCCN=c1ccnc(N2CCOC(c3ccc(Cl)cc3)C2)[nH]1)OC C1(CNC(C2C=CC=CC=C2)=O)CCCCN(C(C2CCOC2C(F)(F)F)=O)C1 c1(CNC(c2[nH]nc(C3CCCN(C(C=CSC)=O)C3)n2)=O)cc(C)ccc1O CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC1CCN(C(=O)Cn2cccc2)CC1C C1(CC)(CO)CCN(C(=O)CCc2csnn2)CC1.C1(C(=O)OC)CCC1C(=O)N C1(C)(CNC(CC2CN(C(C)=O)C2)=O)CCCN(C(c2cccn2C(C)C)=O)C1 c1(OC)cc(OC)nc(C(N2CCC(C(C)NC(=O)CCCC3CC3)CC2)=O)n1 c1(OC)ccc(CNC(C2CC2Cc2c(C)nn(C(C)C)c2C)=O)c(Cl)c1 c1(OC)cc(CC(=O)OCC(=O)C2CC2C(=O)O)ccc1C C1(C(=O)NCCNc2c(C)ccnc2)CCC(C)C(C)C1 C12(C(=O)NCC(CC)(C)C)CCC(CC1)N(C(=O)C(C)C1CCC1)C2 C1(NC(=O)CC2CC2)CCS(=O)(=O)C12CN(C(=O)CC1CCn3cncc3C1)C2 Cc1nn(C)c(Cl)c1C(=O)NC1CCCCC1NC(=O)CC(=O)NC1CC1 c1(OC)cc(C(N2C(C)C3CC2C3NC(=O)CC(F)(F)F)=O)c2occc2c1 C12(C(N(C)CC3CN(C(=O)CNC(=O)CN(C)C)CCO3)=O)CCCC1C2(F)F c1(C(N2CCCN(C(CCC)=O)CC2C)=O)cc2cc(C)cc(Br)c2o1 C1(CN(C(=O)C(Cc2ccccc2)C2CC2)C)C2CN(C(c3ncn(C)n3)=O)CC12 Cc1cc(N2CC(C(N)=O)C(C(F)(F)F)C2)nc(=NCCc2cncs2)[nH]1 N1(C(c2cnoc2C2CC2)=O)CCN(C(=O)CCc2cocn2)C(C2CC2)C1 N1(C(CCONC(=O)OCC)=O)CCN(C(=O)Cc2n[nH]c(C)n2)CC(O)C1 c1(SCC)ccc(-c2nc(-c3nccs3)nn2C(C)CO)cc1 c1(C(=O)NCC(C(=O)N(C2(CCO)CC2)C)CC2CC2)cc2n(n1)CCO2 c1(C(N2CC(CNC(C3CCSC3)=O)C(C(F)(F)F)C2)=O)c(F)ccc(F)c1F C(=O)(CC(C)C(C)(C)NC(=O)C(C)C1(O)CCC1)NCc1c(CC)nco1 c1(CCCC)nc(CN2CC(F)CC2CN2CC(NS(C)(=O)=O)C2)c(Cl)[nH]1 Cc1nc2cncc(C(=O)NCC(C(C)(C)C)NC(=O)CC3CCC(O)C3)c2[nH]1 c1(C(N2CCC(CN(C(C(C)S(C)(=O)=O)=O)C)C2)=O)c2ccccc2nn1C c1(C(=O)NC2(CC=C)CN(C(=O)CSCC3CCCCO3)C2)cc(C)sc1C O=C1CCC(C(=O)N2CCCC(Nc3nccnc3F)C2)=NN1 C12(C(N3CC(O)(CCNC(C45CCCCC4C5)=O)C3)=O)CCCN(CCC1)C2 C1(C(N(CCC#C)CCOC)=O)CC(O)(C(C)(F)F)C1 C(CCCCC(=O)N1CCCC1C(C)(C)COCC)O.C(=O)(C(F)ON=C(C)C)CC c1(CNCC23C(CN(C(C(n4ncc(C)c4)C)=O)C2)C3)cc(O)ccc1Cl c1(C(C(=O)NCC=C)N(C(C)C(=O)OC)CC(C)C)nn(CC)cc1Br CCCC(C)(O)C(=O)N1CC2CC1C2NC(C1CC12CCC2)=O N1(C(Cc2ccn(CC)n2)=O)CCC(C(N2CC3C=CC3C2)=O)C1C(C)C C=C1CCC(C(=O)NCC2(C(=O)NCCC(N)=O)CCCO2)CC1 C1(CNC(COc2c(OC)cccc2)=O)CN(CC(=O)N(C)C)CC12CCC2 C(=O)(CCCC(C)(C)C)NCCC1CN(C(C2(CC)CC(C)(C)C2)=O)C1 c1(OCC(=O)N(C2CCN(C(=O)C(F)=CC3CC3)C2)C)cccc(CCO)c1 Cn1ncc(C(=O)NC2CC3C(NC(C4CCC(C(F)F)CC4)=O)C3C2)c1Cl C1(NC(CCc2nnc(C)s2)=O)CCCC(Nc2ncnc(=N)[nH]2)C1 C(c1ccc(Cl)cc1)=CC(=O)NCC(C1CC1)NC(CCNC(C1C(C)C1)=O)=O C12(CC(=O)NCC(c3ccccc3F)NC(CSCC)=O)COC(C)(C1)C2 C1(C(=O)NC(CNC(=O)C=Cc2ncc[nH]2)C2CCC2)CCc2nnnn2C1 C1(CC(=O)NCC(C)(C)OCCNC(c2c(OC)nsc2)=O)CCCNC1=O C(=O)(C(C)(C)CN(C)Cc1ccccc1)NC(C)C(=O)Nc1nccn1C(F)F N1(C(C2(CC=C)CC2)=O)CC2CC(C1)N(C(=O)C(C)CC(C)(C)C)C2 C(=O)(CCC(C)C)NCC1OCC(C(N2C(C)(COC)CC2)=O)C1 C1(CN(C(CNS(CC)(=O)=O)=O)C)CCCN(C(c2cnn(C3CC3)c2Cl)=O)C1 N1(C(c2c(CC)cc(N)cc2)=O)CCN(C(C2CC(SC)C2)=O)CCC1C C1(CC(=O)NCc2cccc(NC(C(CC)n3ccnc3)=O)c2)CCN(OC)CC1 CCC(CC)C(C)C(=O)NCC1(C2CC2)CCN(C(C2CCOC2)=O)C1 C(C(C)(C)C#CC(=O)N1CCC(CO)C(O)C1)NC(COC(CC)(C)C)=O C(=O)(C1=CCCCCC1)N1CCCC(CCC(=O)N2CC(n3ccnn3)C2)C1 c1(CC)nc2c(C(=O)Nc3cc4nncn4cn3)ccnc2[nH]1 C1(CC)C(NC(c2ccc(SC)s2)=O)CCCN1C(=O)C=CC1CCOC1 C(=O)(CCCCCCSC)NC(C(=O)NC(CC=C)C(=O)OC)CO C1(CC=C)(C(N2CC(O)(C(F)F)C2)=O)CCCN1C(C12CCC(C1)C2)=O N1(C(c2c(OC)nccn2)=O)CC2(C1)CN(c1ccnc(C)n1)C2 N1(C(c2cnc(CC)s2)=O)CC2(C1)CN(C(=O)CC1CC(OC)C1)C2 c1(CC(=O)NCC2N(C(C(C)SC)=O)CC2)ccnn1C C1(C2CC2)(CNC(c2ccnc(CO)c2)=O)CCN(C(=O)C(=O)C(F)(F)F)C1 N1(C(C(C)N(C(=O)CC(C)CNC(C)=O)CC)=O)CCOC(C)(C)CC1 c1(OC)cccc(O)c1C(=O)NC1CC1CNC(=O)C(O)CCN(C)C C(=O)(CCC(C)NC(c1cnn(C)c(=O)c1)=O)NC1C(CCOC)C1 C#CCC(C)(C)C(=O)NCC1C2CCC(C2)N1C(=O)CNC(C1CCOCC1)=O CC1(NC(=O)C2CC2)CCN(C(C23CCC(CO2)C3)=O)CC1 C1(CCC(=O)N(CC=C)CCO)CCC(NC(=O)C(C)Cn2ccnc2)C1 c1(C(N2CC(COC)C(C)(C)C2)C(=O)NCCC2(C)CC2)nc(Cl)cc(Cl)c1C c1(C(N2CCC(O)(CNC(CCNS(CC)(=O)=O)=O)C2)=O)cccc2sncc12 C1(N(C(CN(C2CCCC2)CC)=O)CC2CCCCN2)CCS(=O)(=O)C1 CCC(O)(CC)CCNC(C1CC(NC(c2sccc2C#N)=O)C12CCC2)=O C1(C2CCOCC2)(NC(C(COC)C)=O)CC1.c1(C2C(=O)N2)cnn(C)c1 c1(C(=O)NC2CCC(NC(C3CS(=O)(=O)CCO3)=O)C2)ccc2sccc2c1 CCC(CNC(=O)CC=CCNC(c1cc(C(C)(C)C)n[nH]1)=O)(CC)OC C1(NC(c2nnnn2CCCC2CC2)C2(SC)CCC2)C2CCCOC12 C1(NC(C2CCC(=C)CC2)=O)CN(C(c2ccsc2C#N)=O)CC1N=[N+]=[N-] C(=O)(CCC(F)(F)C(F)F)NCC1CCCN(C(C(C)NC=O)=O)C1 n1(CC(=O)NCC2C(C(=O)NCC3(C)CCC3)C2)cnc(=N)[nH]1 c1(C(N2CC3(CN(C(CS(CC)=O)=O)C3)C2)=O)cc(C)c(C)c2ncccc12 C12(COC)CCCN(N3CC(C4(CC4)C3)OC1=O)C2.C(C)(C)(C)OC N1(C(CNS(CCC)(=O)=O)=O)CCC(C(=O)Nc2cccc(C)c2)C(C)(C)C1 C#Cc1cccc(C(=O)NC2CCCC2N(CC)NC(=O)C(=O)NCC=C)c1Cl C#CC1(O)CC(C(=O)NC(C)C(C)(C)NC(=O)C(C)OCc2ccncc2)C1 c1(C(=O)NC(C(C(C)C)NC(COCCC)=O)C)ccn2ncnc2c1 c1(CC)c(C(=O)NCC(O)CN(C(=O)C(C)N2CCC2)C)csc1C C1(NC(C(C2CC2)SC)=O)C2CC1N(C(=O)CCCc1nc(C)no1)C2C c1(C(=O)NCCC(C)NC(C2CNC(=O)N2)=O)cc(Br)c2[nH]nnc2c1 C1(SC)CCCNC1.C123CC(C1C2)n1cc(nn1)C3.C1(C(F)(F)F)(C(=O)N)CC1 C1(CNC(c2cc(F)ccc2Cl)=O)CC2(CCOCC2)CN1C(c1cncs1)=O C12(CNC3CCCN(S(C)(=O)=O)C3)CCCC1CCO2 n1(CC)cc(CC(=O)NCC(F)(F)CSc2ocnc2C(=O)NC)nn1 Cn1cc(C=CC(=O)NC(Cn2cncn2)C(=O)NCCc2nccn2C)nn1 C1(NC(c2sc(C)c(C)c2C)=O)(CNC(=O)C(N)=O)CC2CCC1CC2 c1(C(N(C)CC2CC2)=O)cnc(CNC(=O)C(C)(C)Cl)nc1.C1(=O)CN1 CC1NC(=O)CCC1NC(=O)CC1(C)CCN1C(=O)Cn1cncn1 C(=O)(CC(C)(C)C(C)=O)N1CCC(C(N(CC(CC)C)C)=O)C(C)C1 N1(C(C2(C#C)CC2)=O)CC2(C1)CN(C(=O)CC1CCN(C)C1)CC(C)(C)O2 C1(NC(CNC(CCC)=O)=O)CC(CO)N(C(=O)Cc2ccccc2C)C1 C1(=CC(=O)NCCC2(OC)CN(C(=O)C(O)CN(C)C)C2)CCN(C)CC1 C1(CCO)(OC(=O)NCC2CCCC2NCc2ccc(F)cc2)CCSCC1 C1(C(N2C(C)(CNC(=O)CCC3OCCO3)CCC2)=O)CCC2(CCOCC2)C1 C1(NC(CNC(CC)=O)=O)CN(C(C2CCCO2)=O)CC2(CCC2)C1 Cc1ccc(NC(=O)CC2CC(F)CN2C(c2ccc(O)c(F)c2)=O)c(O)c1 C(CCCCCNC(=O)CSc1nccn1C)N(C(c1c(C(C)C)scn1)=O)C N1(C(C(CC)N(C)C)=O)CC2(CNC(=O)C=Cc3scnc3C)CCC1CC2 N1(C(C(=O)N(C)Cc2cc(OC)no2)=O)CCc2c(C)cc(Br)cc2C1 C(CC(C)(C)C(=O)NC1CCCN(C(c2ccc(F)c(O)c2)=O)CC1)OC C1(C(=O)OC)CC(C)N1C(=O)CC(C)C1CC1 Cc1cc(CCNC(=O)C(O)CNC(=O)CSc2cn[nH]c2)nn1C N1(C(C(CC)SC)=O)CCOC(CCNC(=O)CC2(O)CC2)C1 N1(C(c2ncn(C)c2Cl)C(=O)NC(CC)C)CCCC12CCCC2 C12(CNC(CC=CCC)=O)CCCCC1CN(C(c1coc(C(N)=O)c1)=O)C2 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)C1OCCN(C(Cc2c(C)nccc2)=O)C1 C1(C)(C(=O)NC(C2CN(C(c3nnc(O)cc3O)=O)CCO2)C)C(C)(C)C1(C)C CC#CC1CN(C(=O)CC2CCN(C(=O)C(C)(C)CSC)CC2)C1 C(c1ccc(Cl)cc1F)=CC(=O)NCC1C(C)(C)C(NC(c2cncs2)=O)C1 N1(C(=O)Cc2ccc(F)c(Br)c2)CCC2(CCN(c3ncc4[nH]ccc4n3)C2)C1 C12(NC(C3C4CCCCCCC34)=O)CCCC1N(c1ccnc3ncnn13)CC2 Cc1cnc(N2CCCN(C)C2)c(S(=O)(=O)NCCS(=O)Cc2ccccc2)c1 c1(C(N(CC(O)CNC(C23CC(C)(C2)C3)=O)C)=O)cccc(C(N)=O)n1 c1(C(=O)NC2CC3CN(c4ccnc(COC)n4)CC23)cc2ccc(Cl)cc2o1 Cc1cccc2oc(=NCc3c(C)nn(CCCl)c3C)[nH]c12 C(Cc1ccccc1)(C(=O)NCCN(C(C1OCC1(C)C)=O)C1CC1)OC C(=O)(C(C)(C)C(F)(F)F)NC(CNC(c1cn(CC(CC)O)nn1)=O)CO C1(C(=O)NC)C=CC(NC(C2CC(CNC(=O)C(=O)NC3CC3)C2)=O)C1 C1(C(N2C(C3(N(C)C(C4CC(O)C4)=O)CC3)CCC2)=O)CCC(O)CN1C N1(C(CC2(C)CC2)=O)CC(NC(C2CCCC(O)C2)=O)CC2(CC2)C1 c1(CCC(N2C(C)(CNC(CN(C3CC3)CC)=O)CCC2)=O)c(F)cccc1Cl c1(C(=O)NCC2C(NC(C3CCC(=C)CC3)=O)C2)ccc(F)cc1C(F)(F)F N1(C(CN(CC(C)C)C(C2CC3CC3C2)=O)=O)CCCC(CC(N)=O)C1 c1(C(N2CCC(NC(C3CCCC3)=O)C2)=O)cc(C(F)(F)F)ccn1 c1(NC(C2CC23CN(C(c2ccc(Br)c(F)c2)=O)C3)=O)ncc(I)cc1[N+](=O)[O-] N#Cc1cc(C(=O)NC2CN(C(c3ccns3)=O)CC2C(F)(F)F)cc(O)c1 CC(C)(C#N)CCCC(=O)NCC1CCCC(NC(=O)C(C)(C)N2CCCC2)C1 N1(C(C2CC(CC)C2)=O)CCC2CCN(C(=O)C=C(C)c3ccccc3C)C2C1 Cc1nn(C2CC2)c(Cl)c1C(N1CCC(CF)(NC(=O)COCC(F)F)C1)=O C(C1=CCN(C(C2(CCN(C)C)CC2)=O)CC1)NC(C1CCC(OC)C1)=O C#Cc1cccc(C(=O)NC(CN2CCN(C(=O)CN(C)C(N)=O)CC2)C)c1 N1(C(C(CC)O)=O)CCn2nc(C)c(CNC(c3cc(=O)n(C)o3)=O)c2C1 C12(CNC(C3(NC(N)=O)CC3)=O)CCC(NC(c3ccnnc3O)=O)(CC1)CO2 N1(C(CS(CC)=O)=O)CCC2CCC(NC(c3cc4cscc4s3)=O)C1C2 CC(C)CC(C(=O)N(CC(O)CNC(C1CC(C(=O)O)(C(F)F)C1)=O)C)C(N)=O Cc1nc(NCc2cc(CC3CC3)no2)cc(=NCC2CCCCN2C)[nH]1 N1(C(C2CCN(C(C(CCC)OCC)=O)C2)=O)CC2(CCC2)OCC1C CC1CN(C(=O)C(O)CC2CCCC2)CCN1C(=O)Cc1cc[nH]n1 Cc1cc(O)ncc1C(=O)NC1CCN(C(=O)CCCc2nncn2C)CC1F C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)CCc2cn(C)nn2)CCC1(C)C c1(C(=O)NCCOCC(=O)N(CCC#N)C2CC2)cc2[nH]ccc2cc1Cl C1(NC(=O)CNC(=O)C2CC2)CCN(C(c2occ3c2CCC3)=O)CC1CO N1(C(C2CC(C(C)C)OC2)=O)CC2CC(C1)N2C(=O)C1CC1 Cc1cc(CCNC(C2CN(C)C(C)CO2)=O)c2ccccc2n1 N1(C(C23OCC(COC)(C2)C3)=O)CCC(CNC(=O)CN(C)CCO)C12CCC2 C=C1CC(C)(C(=O)NC(C)CC2CN(C(C3COCCO3)=O)C2)C1 C1(C2CCN(C(=O)CCc3cnc[nH]3)C2)(NC(=O)CCCc2cnn[nH]2)CC1 c1(OC)ccc(C(N2CCC(C(F)C(N3CCNCC3)=O)CC2)=O)c(Br)c1 C(=O)(C1=CCCC1(C)C)NCC1(F)CC(NC(C2CN(C(C)C)C(=O)C2)=O)C1 Cc1sccc1NC(=O)C(C1CC1)NC(=O)CC1CCCCO1 c1(C(=O)NC2CN(C(c3c(C)c(=O)cc[nH]3)=O)C2)cc2nnn(C)c2s1 C1(CNC(c2nc(CC)oc2)=O)CC(O)C(O)CC1C(=O)NCCCC(N)=O C(CC(C(=O)NC(c1cccc(Cl)c1)CNC(=O)CCC1(C)CC1)NC=O)SC C1(c2cccc(OC)c2)CN(C(=O)C(=O)OC)CCN1C(c1ccc(Cl)cn1)=O C1(C(N(C(CCNC(CN(C(C)C)C)=O)C)C)=O)CCc2cc(F)ccc2O1 N1(C(C(CSC)NC(=O)CC(CN(C)C)CSC)=O)CCn2c(C)nnc2C1 O=C1CC(C(=O)Nc2ccccc2NC2CCC(O)C2)c2ccccc21 C(C(CC(F)(F)F)NC(=O)C(F)(F)C(F)F)NC(C1CN(CC)C(=O)CC1)=O O=C1NC(=O)C2(CCCC2C(=O)NC(c2cccnc2)C2CCC2)N1 C(CCC1CC1)(C(=O)NCC(CC)CCO)NC(C(C)=CC)=O CC1CN(C(C2C3CN(C(=O)CCc4cccc(O)c4)CC23)=O)CCC1=O N1(C(CNC(CC)=O)=O)CCC2(CC1)C(OC)CC2NC(c1ncn(C)c1C)=O Clc1ccccc1-c1ccc(C2CCN(Cc3cc(C4CC4)no3)CC2)cc1 Cc1ccc2occ(C(=O)NC(C)C(CO)NC(C3CN(S(N)(=O)=O)C3)=O)c2c1 C(CN=c1nc(C#N)[nH]cc1Cl)=CCNC(C(CC)C(C)O)=O c1(C(=O)NCC2CN(C(C3CCCC3O)=O)CCO2)ccn2cccc2c1 c1(N2CC(CC)N(C(c3ccc(Cl)nc3Cl)=O)CC2)ncnc2n[nH]c(Br)c12 N1(C(c2ccc(NC)cc2)=O)CCC(CNC(=O)CC2CCCS2(=O)=O)C12CC2 N#Cc1ccccc1C1(CNC(=O)CNC23CCCNCC2C3)CC1 c1(C(c2n(CCC)nnn2)NC2CCSC2)cccc(-c2cccc(F)c2)c1 C1(C(=O)NC2CC(O)C2(C)C)CCC2(CC1)CC2.c1(CC)ncccc1C(=O)OC C(=O)(CCCCCN(C)C)NCC(C1CC1)NC(C(COC)N(C)C)=O CCCCC(O)C(=O)N1CC(NC(=O)C(F)F)C(C)(C)C1 C#CCC(C)(C(=O)Nc1ccc(F)c(CC)c1)NC(C1CCOC1(C)C)=O C1(C#N)(O)CCN(C(=O)COC(F)F)C1.c12cccnc1NC2=O.CC(C)C N1(C(C(CC(F)F)NC(C(C(C)(F)F)F)=O)=O)CCC(C2CCCC2)C1 Cc1ccc2cc(CNCC(=C3CCN(C(=O)C(N)=O)CC3)F)ccc2n1 c1(C(N2CC(O)(C(C)NC(C(C)c3ccco3)=O)C2)=O)ccc2ncsc2c1 C(=O)(CCCC(=O)NC(C1(NC(C2CCOC2C(C)C)=O)CC1)C)NCC Cc1cc(CN(C)C(C2CC2NC(c2ccn(-c3cccnc3)n2)=O)=O)no1 Cc1cc2[nH]c(C(N3CC(O)CC3CC(N3CC4CCOC4C3)=O)=O)cc2o1 c1(C(=O)NCCNC(CC(C)C2CCCO2)=O)cc(Cl)cc(Br)c1 C1(C(N(CC(C)O)CC(N2CCCC2)C)=O)CCCC1CNC(=O)OC(C)(C)C c1(C(N(C(c2cn(CCN3CCOCC3)nn2)C)C)=O)cnn2c1OCCCC2 C1(CNC(C(C)(C)OC)=O)CCCC(CNC(=O)Cc2nonc2C)C1 CCCC(C)(CCC)C(=O)NCC1CC2CCC(C1)N2C(=O)C(CC)OC C=C(C)CCCC(=O)NC1CC(C(=O)NCC(CC(C)C)OC)CC1O C(=O)(C1=CC2(CCOCC2)C1)NC(C(C)NC(CCC1CC(OC)C1)=O)CO CCC(C)C(C)CNC(C1(C)CN(C(C2(n3cccn3)CC2)=O)C1)=O C1(O)(CNC(CCNC(C(C)(C)C2CCC2)=O)=O)CCCC1(C)C N1(C(c2c(C)nc(C)s2)=O)CC(=O)NCC1c1ccccc1 C12(CNC(C3CCN(C)C3)=O)CCC(CN1C(c1ccc(SC3CC3)nc1)=O)C2 N1(C(c2cccc(SCCC)c2)=O)CCC(NC(=O)C(F)=C2CCC2)CC1C N1(C(CCOC)=O)CCn2ncc(CNC(C34CCC(CC3)CO4)=O)c2C1 C(=O)(C(F)C(C)CNC(c1sccc1F)=O)NCc1cc(OC)ncn1 N1(C(COCC)=O)CC(NC(=O)C(F)C(F)(F)F)CC12CCC2 CN1CCCCCC1c1nnc(NCC2C(O)C(O)CN2C(=O)OC(C)(C)C)[nH]1 C1(C(N2CC3C(C)(C)C3C2)=O)CCN(C(C2(OC(C)C)CCC2)=O)CC1(C)C c1(OCCNC(C2C(C(=O)Nc3n(CC)ncc3)C2)=O)ncc(C)cc1Br c1(C(N2CC(F)(C(N(CCOC)CCO)=O)C2)=O)cc(N)cc(F)c1 N1(Cc2ccc(OC)cc2)C(=O)NC2(CCCCC2C)C1=O CC1CCOC1CC(N1CCCC1CC(=O)NCC=CBr)=O c1(CC(=O)NC2CC(NC(C(Br)=C(C)C)=O)C(O)C2)cccc(C)c1C C1(C(=O)NC(C#C)CC2CCC2)(CNC(=O)CCC2CCCO2)CC12CCC2 C1(NC(C=COCC)=O)CCCN(C(c2ccc(-c3ccc(O)nn3)cc2)=O)C1 C(=O)(C(C)(C)C(O)C(C)C)NCCCCC(=O)NC(COCC)CO N1(C(C2C(c3cc(C)sc3)C2)=O)CCCCC1C(C)(C)CNC(c1ccon1)=O c1(C(=O)NC(C2(O)CN(C(=O)COC3CCCOC3)C2)C)ccnc2[nH]ncc12 C1(CCNC(C=COCC)=O)CCCN(C(=O)CC2CCCO2)C1 N1(CC)CC(C(=O)NCc2cc(C(N3CC(CCO)C3)=O)cs2)CC1=O c1(C(=O)NC(CCCNC(c2c(CC)nn[nH]2)=O)C)cccc2cnn(C)c12 c1(C(=O)NC2(C)CCN(C(C3CC(C(=O)OC)C3)=O)C2)coc2ccc(C)cc12 N1(C(C(C)CO)=O)CCOC(C(C)NC(c2ccccc2C2CCCC2)=O)C1 C(N=c1[nH]cnc2c(OC)cccc12)C1CCN(C(C(COCC)N=[N+]=[N-])=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CCCCC(CCC(=O)NCC(=O)OC(C)C)C1 C12(C(=O)NCC3N(C(c4c(Cl)cn(C)n4)=O)CC4(CC4)C3)CCCCC1OCC2 C1(C(N)=O)CC12CCN(c1cncc(NC3CCC3)n1)CC2 C1(C)(COC)CC(NC(c2cn[nH]c2)=O)CN1C(C1CC(F)(CF)C1)=O N1(C(CCN(CCCC#C)CC)=O)CCN(C)C(CNC(=O)C(O)CC(N)=O)C1 C1(CNC(C(CC#C)C)=O)CCN(C(=O)CCSCc2ccccc2)CC1(F)F C12(NC(c3csc(-c4ccccc4)c3)=O)CC1CN(C(C1(CO)COC1)=O)C2 C1(C(C)C)(C(=O)N(C)CCN2CCCC2)COC1.C1=CCNC1=O c1(CNC(CC2(CNC(C=Cc3cc(C)no3)=O)CC2)=O)ccc(C)c(C)n1 C(CCCC(=O)NCc1ccnnc1O)OCCC=C c1(C(=O)NCC(CC=C)NC(=O)CCC(F)F)ccccc1C(=O)NC(C)(C)C C1(C(N2C(C)(C(=O)OC)CC2)=O)C2CCCC2CN1C(=O)Cc1ccon1 C12(CC=CCC1)C(=O)N(C)C2.N1(C(C(C=CCCC)O)=O)CCOC(CCC)C1 Cn1c(NC(C2(C)CCCN(C(c3ccncn3)=O)C2)=O)cc(O)nc1=O c1(C(N(CC(CC)NC(=O)C(C)(C)c2ccn(C)n2)C)=O)n[nH]cc1C1CCC1 N1(C(C2C(CC(C)C)C2)=O)CCC(C)(C(=O)NCC2(C)CSC2)CC1 C(=O)(C1=CCOCC1)NCCC1CCC(NC(C=C2CCN(C)CC2)=O)C1 C1(C(N2CC(C)(NC(CC=CC=C)=O)C2)=O)CCCC1C1CC1 C1(C(N(C2CN(C(=O)CCCc3ccncc3)C2)C)=O)CCS(=O)(=O)N1 C(N=c1[nH]c(N(CC(c2ccccc2)C)C)nc2c1CCCC2)c1ncc(C)cn1 N1(c2ncc(C)c(-c3ccccc3)n2)CC2CC1CCC2NC(=O)C1=CCSC1 N1(C(c2c(OC)ccc(C)n2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 CC1CCC(CC(N2CCCC2Cc2cn(Cc3cccc(O)c3)nn2)=O)CC1 C(C(C(=O)NC1CN(C(C2C3CCC(F)(F)C23)=O)C1)C(C)(C)C)OCC=C CN=c1[nH]cc(C(=O)N(C(C)CNC(C2CC2(c2ccccc2)C)=O)CC)o1 C1(C(N(C(=O)CN2CCCC2CNC(=O)N(C)C)CC)=O)CN(C)CCO1 C1(C(=O)Nc2cnc(Cl)c(Cl)c2)CCc2nc(-c3cccc(O)n3)sc2C1 C12(c3cn(C(CNC(CC(C)c4cnn(C)c4)=O)C)nn3)CCCC1CC(=O)C2 N1(C(C(CCC#C)NC(=O)C=C(C)C)=O)Cc2cccc(F)c2C1 C(C)(C)(CC(C)(C)C)NC(CC1CCC(NC(C2C(C(C)C)OCC2)=O)CC1)=O c1(C(=O)NCCC2CN(C(C3(CC)CC3)=O)CC2C)cc(=O)c2ccncc2o1 c1(C(=O)OC)cccc(C)c1Nc1cc(C)nc(C2CCCO2)n1 C1(NC(CCCCOCC)=O)CN(Cc2csc(C)n2)CCC1C C(CC1=CCN(C(c2nnn(C)n2)=O)CC1)NC(C1N(C(C(C)C)=O)CCC1)=O C(C(O)C(=O)N(C(C)CCN1CCCC1)C)SC.C1(=O)C(NC(C)=O)CN1 C(c1c(Cl)cccc1Cl)=CC(=O)NCCc1cc(C)on1 C1(C(=O)Nc2nc(O)cc(C(=O)OC)n2)CCCC2CCCCC12 C(=O)(CCCC(=O)NC1CS(=O)(=O)CC1NC(=O)C(F)(F)c1ccccn1)OC C1(C(N2C(c3nnc(C)o3)CC3(CCC3)C2)=O)CCc2nnn(C3CCC3)c2C1 CC1CCC(CNC(C2(C)CC2)=O)CN1C(c1coc(C(F)(F)F)c1)=O O=C(C#CC1CCC1)NCC12CC1CN(C(=O)CCC1CCC(C(F)(F)F)O1)C2 N1(C(c2c(C)ncs2)=O)CC2(CNC(=O)C(c3ccccc3Cl)(C)C)CC1CO2 C(N=c1[nH]c(=NC)[nH]c(=NCC(CSC)SC)[nH]1)c1ccc(OC)c(Cl)c1 C(=O)(C(N=[N+]=[N-])C(C)C)N1CC(CCC=C)(C(N2CC3CC3C3CC23)=O)C1 C1(C(N2C(C)CC(NC(=O)CC3CCCC3)C2)=O)CC2(C1)CC(F)(F)C2 C1(N(CC)CC)(C=CC(=O)NC)CCN(C(=O)CS(=O)(=O)NC2CCC2)C1 N1(C(C(=O)NC2CCCO2)C2C(OC)C2)CCC2CC12 N1(C(c2c(C)onc2O)=O)CCC2CCC(C1)N2C(=O)C(=O)N=S(C)(C)=O C1(CNC(C=COCC)=O)CCCC(CNC(c2cnn(C3CCC3)c2)=O)C1 CC1(NC(C2CC3CC3C2)=O)CC(NC(c2ccsc2-n2cnnn2)=O)C1 Cc1nc2c(C)cc(C(N3CCOC(CN(C(=O)C(C)CO)C)C3)=O)cn2n1 N1(C(C2CCN(CC)CC2)=O)CCC(C2CC2)C1C(N1CC(OC(=N)O)C1)=O CC(C)(C(=O)NC1(C)CCCOC1)C1=CCN(C(c2cc[nH]n2)=O)C1 CCCC(CCC)CN=c1cc(C)[nH]c(=NCc2ccnc(C)c2)[nH]1 C(=O)(CC(C)C(F)F)NCC(C)CN(C(=O)C(F)(F)C(O)C1CC1)C Cc1ccc(SCCC(=O)NC2CC(OCCNC(=O)C(C)C3CC3)C2)c(C)c1 c1(C(N(CCNC(C(CC=C)Cc2ccccc2)=O)CC)=O)ccc(N)c(Cl)c1O N1(C(C=Cc2ncn(C)c2)=O)CCN(C(c2n[nH]cc2C(F)(F)F)=O)C2CC12 C1(O)(C(N)=O)CCN(C(=O)CCC2CCN(C(C3(Cl)CC3)=O)CC2)CC1 c1(NC(C)=O)ccc(OCC(=O)OCC2CCCO2)c2ccncc12 C(=O)(C1=C(C)CCC1)N(C(C(=O)N(C)CC1(COC)CCC1)C)C1CC1 CCC(=O)NNC(=O)C(C)OC(=O)Cc1cnn(C)c1C C1(C(C(=O)NCCOC)N(C)Cc2ncnn2C)CCCOC1 c1(C(=O)NC2CCC(N(C(CS(=O)(=O)NC)=O)C)CC2)ccn2c1CCCC2 Cc1nnn(CC(=O)N(CCC(C)NC(C2(CO)COC2)=O)C)n1 c1(CC(N2CCC(NC(C3C(=C)C3)=O)(COC)CC2)=O)sc2ccccc2c1C C1(CC(=O)NCC(O)CNC(=O)CC(F)(F)F)NC(=O)CNC1=O c1(CN2CCCC(C(C)NC(c3nc(C)nn3C)=O)C2)c(F)cccc1F N1(C(CCOCCOC)=O)CC(NC(C2(NC(N)=O)CC2)=O)C(C)C1 CC1CN(C(C23CC2CCN3C(=O)Cc2ccc(F)cc2)=O)CCS1 C1(C(=O)NC23CC(CNC(CSCC(=O)OC)=O)(C2)C3)CCN(C)C(=O)C1 C1(NC(c2nc(C)sc2C)=O)CCC2(CC1)CN(C(=O)Cc1cnc[nH]1)CCO2 n1(CC)cc(C(=O)NC2C=CCN(C(c3cc(OC)ns3)=O)C2)c(C)n1 Cc1cc(C)n2nc(C(=O)NCC3COCCN3C(c3ccc(F)o3)=O)cc2n1 C1(C(N(C(CC)CO)CC)=O)CC2CN(C(c3nccs3)=O)CC2C1 n1(CCC)nc(C2CC2)nc1C1=NOC2OCCCC12 N1(C(CC2(C)CC2)=O)CCCC(NC(C2Cc3nncn3C2)=O)CCC1 N1(CC#C)CCN(C(=O)C(O)CNC(c2sccc2C)=O)CC1=O c1(C(N2CCCC(N(C(=O)COC3CCC3)CC)C2)=O)cc2ccncc2s1 C(=O)(C1=CCC2CCC1N2C(C1CCC(C)(C)OC1)=O)N(CC(C)O)CC(C)O N1(C(CCC)=O)CCC(N2CCCC2C(=O)Nc2ccc(OC)cc2)CC1 C=C(C)c1cn(CC(C2CN(C(=O)CCOC(=O)C=CCOCC)C2)F)nn1 CCCS(=O)(=O)C1CCCC1C(=O)NCC1CCN(C(=O)Cc2cnoc2)CC1 N1(c2nc(NC(c3cccc(C)c3)C)nc(C)c2)CCC2(CCCOC2)C1 c1(C(N(CC(C)N(C(c2c(C)cc(SC)o2)=O)C)C)=O)cc(C)cc(C)c1 C1(CNC(CC=CC=C)=O)(NC(=O)C(C2CCCOC2)OC)CCC(F)(F)CC1 CCC(F)(F)CC(=O)NC1CC12CCN(C(=O)C(C)c1ccsc1)C2 C(CCF)(C(=O)NC(C)(C)CCOC)NC(c1c(CC)cc[nH]1)=O N1(C(C(CC#C)O)=O)CC2COCC(C1)C2NC(c1[nH]cnc1CC)=O c1(CC)c(N2CC3C(NC(=O)CN4CCCCC4)C3C2)nc(C)nc1Cl c1(OC)cc(C(N2CCC(NC(=O)C3=CCC3)C(O)C2)=O)c(Cl)cn1 N1(C(c2ccc(C(=O)NC)cc2)=O)CC2(C(=O)Nc3ccccc3)CCC1C2 CC(C)CC(CNC(C1C2CCC(=O)C12)=O)NC(c1ccn(C)n1)=O c12nc(nc3sccc13)[nH]2.Cc1ccc(SCCOCc2cc(C)sc2C)cc1 C(C(C(=O)NCC1CN(CC)C(=O)O1)C(C)C)NC(c1c(CC)non1)=O N1(C(C)C)CCC(N2CCC(CC(=O)N(C3CCCNC3=O)C)C2)C1=O n1(CC(=O)N(C2CCN(Cc3cn(C4CCCC4)nn3)C2)CC)cnc(Br)n1 c1(NC(Cc2cc(OC)c(C)cc2)=O)cc(Cl)cc(Br)c1F C(=O)(C1(C)CCn2c(C)nnc21)NCC1C(NC(CCc2c(C)cccn2)=O)C1 C(C(CC(=O)N(C)CCC(C)C(C)C)C1CCC1)NC(C1(OCC)CCC1)=O c1(C(N2C3(CNC(c4cnc(COC)s4)=O)CC(C2)C3)=O)nccn2ccnc12 c1(C(N(C)CCNC(=O)CC2COCCO2)=O)csc(-c2ccsc2)n1 O=C1CN(C(=O)CS(=O)(=O)NC2CC2)C2CCN(C(C3CCCO3)=O)CC2N1 N1(C(CC2(C)CC2)=O)C2CCCC1CN(C(c1cccc3oc(O)nc13)=O)CC2 N1(C(C(CC#C)O)=O)CC(C2CCCN(C(c3ccc(C)c(C)c3)=O)C2)C1 C1(OC)CN(C(=O)Cc2cccs2)CC1CNC(c1ccnc(C2CC2)c1)=O N1(CC(=O)NCCCN(C(C(C)C2CCOC2)=O)C2CCCC2)CCC(O)CC1 CC1CCN(C(C23CC(CN2C(=O)C2=NOC(C)C2)C3)=O)CC1O N1(C(CCC2CCN(C(COC)=O)C2)=O)CCN(C)CC1C1CC1 c1(N(C(=O)CC2(C)CN(S(=O)(=O)C3CC3)C2)C)ncc(F)cc1I N1(C(C(C2CCC2)OCC)=O)CCC(C)(CNC(c2c[nH]nc2C(F)(F)F)=O)C1 N1(C(C(CC)(CC)CO)=O)CC23CCCC2(C1)CN(C(=O)Cn1cc(N)cn1)C3 N12C(=O)CN(C1=O)CCC(=O)NC(C)C2c1cccc(F)c1.Cc1ccccc1 c1(OC(F)(F)F)cccc(-c2noc(C3C=CCC3)n2)n1 C1(CC)(NC(C23CC4CC2C3C4)=O)CCCN(C(c2cc(OC)ccc2Cl)=O)C1 C12(C(N3C(CNC(CSC)=O)CC(C)(C)C3)=O)CCC(C)(CC1)OC2(C)C Cc1[nH]nc(C(=O)NCC(C)(C2CC2)NC(C2CCCC2C(C)C)=O)c1C CCC(C)CCC(=O)N1CC(N(C)C(C2(C)CC2)=O)C(O)C1 C(CCC(C)C)(C(=O)Nc1ccc(CCCC(=O)OC)cc1)NCCC N1(C(CCC=CC)=O)CCC2(CC1)OCCC2NC(=O)C(C)NC(C1CCC1)=O CC1(C)CC(NC(c2c[nH]c(=S)cn2)=O)CN1C(=O)CNC=O C1(OCC)CCCN(C(=O)C(CCF)NC(=O)CC2CCSCC2)C1 Cc1ncc(C(=O)NC2CN(C(c3cnsc3)=O)CC2C)n1C(F)F C1(C(=O)NC(C)C(C)NC(N)=O)CCCCN1NC(C=C(C)C(C)C)=O C1(C(=O)NCC2CCC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CC(S(N)(=O)=O)C1 N1(C(C(C=C=C)C)=O)CC2(CC2)CC1CC(=O)NCC(c1cccs1)C C(C(C)(C)CC(=O)NCC1CCCN1C(C12CSCC1C2)=O)OC N1(C(C(C)OCCC=C)=O)CCC(C2CC2)(CNC(=O)COc2ccn(C)n2)C1 c1(C(=O)OC)sc(C(=O)NC(C)CCNC(c2nocc2C)=O)cc1C C(=O)(CCCC(=O)C(C)(C)C)NC12CN(C(CCC(C)CC(=O)O)=O)CC1CCC2 C(C(C)(O)CC(=O)NC1C2CN(C(=O)C(c3ccc(Cl)c(C)c3)(C)C)CC12)OC C1(C)(CN(C(=O)Cc2cccnc2F)C)CCCC1NC(=O)C=CC1(C)COC1 C=CCCCCC(C(=O)N)N(C)SC.C1(N)COCCC1(C)C CC1=CCC(C(=O)NCC2(C)CCCN2C(=O)C=Cc2cc(C)no2)CC1 c1(CC)nc(N(CC(C)NC(=O)Cc2cc(C)on2)C)c(C#N)cc1C N1(C(C(CC)C)=O)CCC2(CC(C(N3CCCC(F)CC3)=O)C2)C1 c1(C(=O)OC)ccc(-c2ccc[nH]2)c(N=c2[nH]c(C3CC3)nc3c2CCCC3)c1 C1(C(N(C(CNC(=O)C(C2CCCCC2)O)C2CC2)C)=O)CC(O)(C(F)(F)F)C1 C#Cc1ccnc(C(N2CCC(CNOC(C3CC(C)OC(C)C3)=O)C2)=O)c1 N1(C(c2nc(CCC)oc2)=O)CC=C(CNC(c2cc(Cl)ncc2OC)=O)CC1 N1(C(C(=O)NCCOCC)CC2CCC(C)CC2)CCC(C(F)F)C2(CCC2)C1 C(C)(C)(CCNC(C1CCOC1CNC(=O)C(CC1CC1)OC)=O)OC C1(NC(CCN2CCC(C)CC2)=O)(CNC(=O)CC2(C)CC2)CCCCC1C C#CCC(C)(C)CN(C)C(c1nccn1CC)c1nnnn1C1(C)CC1 C=CC(CC)CC(=O)NCC=C1CCN(CC2CC(C)(C)C2)CC1 CN(C)S(=N)(=O)c1cccc(-c2nc(C(C)(C)C)nn2C23CC(C2)C3)c1 c1(C(N2C(C)CC(NC(C3CC3(F)F)=O)CC2)=O)cc(O)c2sccc2c1 Cc1ccc(Cl)c(C(N2CC(NC(c3n[nH]cc3[N+](=O)[O-])=O)CC2(C)C)=O)c1 C1(CN2CCC(CNC(C(C)OCC3CCCO3)=O)CC2)OCCN(C)C1=O C1(C(=O)NC2(CO)CCCN(C(c3c[nH]c(=NC)o3)=O)C2)CCC([N+](=O)[O-])CC1 C1(C)(CC)CCCN(C(C2(C)CCCN2C(C2CCCC(=O)CC2)=O)=O)C1 N1(C(C2N(C(c3c(OC)ccc(I)c3)=O)CCOC2)=O)CCNCC12CCC2 CC(C(=O)N(C(CNC(C1CC1C(F)F)=O)C1CC1)C)n1cncn1 CC(CC(=O)N(CCCN(C)C(c1cccc(N2CCOCC2)n1)=O)C)C(F)F C1(C(N(CC(C)NC(=O)C2=COCCO2)C)=O)CCCCC(=O)C1 N1(C(C(CC)(F)F)=O)CCN(C(=O)CN2C(=O)CCC2=O)CC12CC2 c1(CCC(=O)NC2CCCC2NC(c2ccc(C(F)F)o2)=O)nnc(O)nc1O c1(C(N(C2CN(C(c3cn(C(F)F)cn3)=O)C2)C)=O)ccn(C)c1 c1(C(C(=O)N(CCCNC(=O)C(C)Cc2ccncc2)CC)C)ccc(C)cc1 C1(CNC(c2ccnc(C)n2)=O)CC2CCC(C1)N2C(=O)CC1CCS(=O)(=O)C1 Cc1ncc(CC(=O)NCCC2CN(C(c3ccns3)=O)CCO2)c(O)n1 C(C(O)CC(=O)N1CC(O)CC1C1CCCOC1)NC(C)=O C#Cc1cccc(C(=O)NCC2(C(=O)N(C)CC3CCCC4CC34)CC2)c1C CC1(C)C(=O)CC1C(=O)NC(C)(C)C=CC(=O)NCC1(C)CCCS1 C1(CNCC(C2CCC(F)(F)CC2)C)C(=O)Nc2ccccc2S1(=O)=O CC(CN(C)C)CCC(=O)N1CCC2C(NC(=O)COCCOCCO)C2C1 C1(NC(c2c(CC)non2)=O)CCOC(C(=O)N(CC)Cc2cn(C)nn2)C1 Cc1[nH]c(C)c(C(N2CC(CNC(C3CCCOC3c3cn[nH]c3)=O)C2)=O)c1C CN=S(C)(=O)c1cccc(C(=O)NCCNC(=O)CC2OCCCC2(C)C)c1 c1(OC)ccc(CCNC(=O)NCc2cn(C)nc2CC(C)C)c(Cl)c1 N1(C(C2N=C(C)SC2)=O)CCCC(NC(C2(S(N)(=O)=O)CC2)=O)C1C C#Cc1cccc(C(=O)NCC2CC(C(=O)N(C3(CO)CC3)C)CO2)c1C CCCC(C)(CCC)C(=O)NC1(CNC(c2nccn2CC)=O)CCCCC1C C1N(C(C2CC3CCC2N3)=O)CCS(=O)(=O)C1 C1(C(C)NC(c2c(C)snc2)=O)CCCN(C(=O)CC2CCN(C)CC2)C1 c1(C(N(C(=O)C(C2CCCCCC2)O)CCCS)=O)cc(C)cc(C)c1O.CC C1(CNC(c2nc(NC(C)=O)sc2)=O)CN(C(=O)C(F)=CCCF)CCC1C C1(C(=O)NC(C(=O)OC)CC2CCC2)CCC2(CC2)N1C(=O)C(C)CN(C)C N#Cc1ncc(C(=O)NC2CCC(CNC(=O)C(C3CCCO3)C3CC3)C2)c(O)n1 c1(CC)cc(C(=O)NC2CC(NC(c3nnn(C)c3C)=O)C2)c(C)o1 C(=O)(C(O)C1=CCCCC1)NC1C(N(C(=O)C2=CCOCC2)C)CC1 c1(N2CC(CC(C)NC(=O)CC3COCCO3)C2)ccn2ccnc2n1 c1(C(N2CC(NC(Cc3c(C)nsc3)=O)C(O)C2)=O)cc2ccc(Cl)cc2o1 C1(CNC(CC2N(C(c3c(C)cc[nH]3)=O)CCOC2)=O)COCC(C)(C)O1 C(C(N=[N+]=[N-])C(=O)NC1(CO)CCCN(C(=O)C(C)C2CCCO2)C1)OCC c1(NC)ccc(C(=O)NC(CO)C(C)NC(=O)CCOC(C)C)cc1.C(CCO)N c1(-c2ccc(CN(c3ccc(CC)cc3)CC)s2)nc(C)c(N(C)C)s1 CCC(O)C(=O)NCCOC1(NC(=O)C(C)Cc2ccco2)CC1 Cc1nc(NCC(C2CC2)N(C)C(C2CC3CCCC23)=O)cc2nncn12 C1(C2CCCCC2)(C=O)CC1.C1(N(C(=O)CCNC(C2CCC2)=O)C)CC(N)C1 C1(OC)CN(C(=O)Cn2ncn(C)c2=O)CC1NC(c1ccc(Cl)o1)=O C1(n2cccn2)(NC(CCOCC)=O)CCN(C(=O)C(CCSC)OC)CC1 c1(COC)onc(C)c1CN1CCC(c2cccc(I)c2)C1 C(C)(CCCCCO)OCCCC(C(C1CN(C(CCOC)=O)C1)O)=O c1(CC(=O)NCCC(CNC(C2CC2C(F)F)=O)OC)ccc(C)cc1C N1(C(C23CC(C#N)(C2)C3)=O)CCC(NC(C2CCc3cncn3C2)=O)CC(O)C1 C12(C(=O)NCC3N(C(Cc4nc(NC=O)sc4)=O)CCSC3)COC(CCO1)C2 c1(C(N(C(CCNC(CC(C)C)=O)C)C)=O)cncc(-n2cccn2)n1 C(C)(C)(C(=O)NC1CCC(C(C)C)C1)NC(=O)NCCC.c12ocnc1C(=O)N2 N1(C(c2c(C)cco2)=O)CCN(C(=O)C2CC2)C(c2cn[nH]c2)C1 C1(C(=O)NCCn2cc(C3CC3)nn2)CCC2CCC1N2C(=O)Cc1nc[nH]n1 c1(C(=O)NCC(CNC(C(C)OCC#C)=O)(C)C)cnc(S)n1C C1(C)(C(N(CCN(C(=O)C(C)(C)C)C)C)=O)CCCN(C(=O)CSCC(F)F)C1 C(C)(CN=c1[nH]cnc(Cl)c1F)NC(c1c(OC)ccc([N+](=O)[O-])c1)=O N1(C(C2C(CC)OCC2)=O)CCN(C(c2ccc(CO)s2)=O)CC12CCC2.C(C)(=O)N N1(C(C2(OC)CCC2)=O)CCC(CCNC(=O)C(F)=C(C)C2CC2)C1 C1(C(N(CCCNC(=O)Cn2cnc(Br)c2)C)=O)CCCC(N(C)C)C1 c1(OC)cccc(CN(C(CCCOC(C2(CO)CC2)C2CC2)=O)C)c1 c1(C(N2CCC3(N(C(=O)Cc4cocn4)C)C(C2)C3)=O)cnc2ccccn12 S(=O)(=O)(C1CCN(C(=O)CCn2cc(Cc3cccc(CO)c3)nn2)C1)NCC C(C(C(=O)NC1(C)CCOC1)C(C)C)NC(c1n(CC)nc(C)c1)=O c1(N(C)CC2(C)CCC2)nc(N(CCCOC(C)(C)C)C)c2ccccc2n1 Cc1sc(O)nc1C(=O)NCCC(C)(C)CNC(c1csnn1)=O N1(C(C23CC(CN(C(C(C(C)C)SC)=O)C2)C3)=O)CCC2(CCCCO2)C1 C(=O)(C1SCCc2ccccc21)N(CC(C)N(C(c1nccc(OC)c1)=O)C)C c1(OC)cc(F)ccc1N1CCN(C(=O)NC(c2cccnc2)CN(C)C)CC1 c1(OC)ncnc(C(=O)NCC(F)CNC(c2cn(CCO)nc2C)=O)c1F N1(C(COc2cccc(C)c2)=O)CCC(NC(C2(C)CCCS2)=O)CC(O)C1 C12(C(N3CC(C)(NC(C4(C)CCCN4C)=O)C3)=O)CCC(CF)(C1)OC2 C1(C)(CNC(C2CN(C(C)C)C2)=O)CCN(C(c2c[nH]nc2-n2cnnn2)=O)C1 Cc1ccc(C(=O)NCC2(C(N3CCCCC3CC(N)=O)=O)CC2)c(F)c1 Cn1cc(S(=O)(=O)NCC2(F)CCCN(C(=O)Nc3cnc[nH]3)C2)cn1 C1(C(N2CC(C)(C)C(NC(C3CCC3(F)F)=O)C2)=O)CN2CCCN1CC2 C(CCC)(CCCNC(=O)CN(C)C)NC(c1nc(CCC)oc1)=O.C1C(=O)N1 C12(CCC)CN(CCC3CCCO3)CC(C3CC3)(C1)C2.c12ccnc(n1)S2 C(=O)(C(O)CC(F)(F)F)N1CC(SC)C(NC(C23CC(CN2C2CC2)C3)=O)C1 c1(OC)ccc(C(C)(C)C(=O)NC2CC(NC(C3CC3C)=O)C(O)C2)cc1OC c1(C(N2C(C(=O)NCC(C)(C)C(N)=O)CC(OC)C2)=O)ccc2c(c1)CCN2 Cc1ncc(NC(C2(C)CCN2Cc2ccnc(F)c2Cl)=O)cc1Br Cc1ccc(=N)[nH]c1C(N1CCC(C)(CNC(C2(C)CC=CCC2)=O)C1)=O c1(C(C)C(=O)NC2CC(NC(=O)CCN3CCCCC3)C2)ccc(F)cc1F C=C(C)C(CC(=O)N1CC(CNC(=O)CC2CCC(F)(F)CC2)C(C)C1)OCC N1(C(CCCC(=C)C)=O)CCC2CN(C(=O)CSCc3ccncc3)CCC2C1 CC(C)(C)C(CNC(=O)CNc1cn[nH]c1)C(=O)NC1CCCC12CC2 C1(C(C)C2CC2)CN(C(C2C=CCN2C(=O)COc2cccnc2)=O)CCO1 C1(CC(=O)NC)CN(C(c2ccc(Cl)cn2)=O)CCN1C(=O)C(C)C1CCC1 C1(C(N2CCC(CCNC(=O)Cn3cccnc3=O)CC2)=O)(OC)CCCOC1 Cn1c(N2CC3C(C(F)F)C3C2)nc2cc(Br)ccc12 N1(C(c2nc(C)oc2)=O)CCC2CC1CN(C(=O)CC1CCCOC1)C2 n1(C(C)C)ncc(CNC2CN(CC)CC2C(F)(F)F)c1F.C(C)(C)(C)OC(=O)O c1(C(=O)NCC2(C)CCN(C(C3CCCC4CC34)=O)C2)c(Cl)oc2ccccc12 CC1(NC(=O)CCc2nnc(C(F)F)o2)CCN(C(C2CC2F)=O)CC1 C1(OC)CC(CNC(=O)C(C)(C)c2ccn(C)n2)N(C(c2cnc(C#N)s2)=O)C1 N1(C(C2C(NC(CN3C(C)CCC3)=O)COC2)=O)CC2CCCC2C1 N1(C(C2CC(=C)C2)=O)CCn2ncc(CNC(c3csc(C)c3C3CC3)=O)c2C1 N1(C(C(C)CC(F)F)=O)CC2=C(C1)CN(C(=O)COCc1ccnn1C)C2 NS(=O)(=O)c1n[nH]cc1C(N1CC(C(N)=O)(CNC(C2(F)CCCCC2)=O)C1)=O C=CC(CCC)CC(=O)NCC1(CNC(C2Cc3ccccc3O2)=O)CC1 c1(C(C(=O)NC)NC(c2nnnn2C2CCCCC2)(C)C)conc1C(C)(C)C N1(C(c2c(C)n(CCO)cc2)=O)CCN(C(c2cncn2C)=O)C2CCC12 C1(CNC(Cc2cc(OC)cc(OC)c2)=O)CCC(C)(C)CN1C(C1CCC1)=O N1(C(C2N(C)CC2)=O)CCCC1C(N1CCC(c2ncc[nH]2)C1)=O C(=O)(C(=O)N=S(C)(C)=O)NCC(C)CN(C(=O)C(c1ccc(F)c(F)c1)(C)C)C C(C)(CC(=O)N1CCC1C1(NC(c2cnc(S)nc2)=O)CC1)(C(F)F)N(C)C C1(NC(Cn2cccc(C)c2=O)=O)CC2CCC(C1)N2C(=O)CN1CSCC1=O C1(C2CCCCC2)(NCCCNC(=O)COc2ccnc(C3CC3)n2)CC1 c1(C(=O)NC2(C(=O)NCCCC(=O)NC)CSC2)cc(C#N)cn1C c1(CCC(=O)N(CC(C)NC(C2CCC(C)(F)CC2)=O)C)ccc(F)cc1F c1(OC(=O)NCC(N2C(C(N)=O)COCC2)=O)ccc2[nH]cc(C(N)=O)c2c1 c1(OC)ccc(Br)cc1C1(C(=O)NCCN(C(=O)C2=CCSC2)C)CC1 c1(N(CCN2CCOC2)C)ccc(Br)nc1[N+](=O)[O-] N1(C(C(C(C)C)NC(COC)=O)=O)CCCCC2(C1)CN(C(c1cnns1)=O)C2 S(=O)(=O)(c1nccs1)NCC1CCC(NC(c2cc(CC)[nH]n2)=O)CC1 N1(C(C(C)=CC=C)=O)C(C(=O)NC2(C(C)C)CCC2)CCC1C(C)C c1(C(=O)OC)ccc(NCC2CCC(OC(F)(F)F)C2)c(C#N)c1 CN1CCc2[nH]nc(C(=O)NCCCCCCNC(c3ccc(Cl)[nH]3)=O)c2C1 c1(C(=O)NC2CC3C(NC(c4ccccc4)=O)C3C2)ccc(F)c(F)c1 C(=O)(C(=O)C(C)C)N1CC(C(=O)NC(c2ncccn2)CC)(SCC)C1 N1(CCOCC)C(=O)NC(C)C1=O.C1(CC(=O)OC)CCCC(C)C1 N1(C(CC)=O)CC(C2CCCN(C(=O)C=C(C)COC)C2)C1 N(C(=NCCCF)NCCF)C(C)Cc1ccccc1 c1(CNC(N(C)C(c2ccccc2Cl)C2CCOC2)=O)ccc2c(c1)CCCC2=O C1(Nc2ccc(C(=O)NCCSCC=C)s2)CCN(C(=O)C2CC2)C(C)C1 c1(C(=O)NC(CN(C(c2ccc(OCC(C)C)nc2)=O)C)C)ccc(F)cc1Cl Cc1nccc(N2CC3CC2C3C(N2CCCC2C)=O)n1 CC1(NC(C2(CF)CC2)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)C1 C1(CNC(CSCC)=O)CN(C(=O)C(c2c(F)cccc2F)C)CC12CCC2 N1(C(Cc2nc(C)oc2)=O)CC2(CCN(C(C3CCCCC3C(F)(F)F)=O)C2)C1 c1(CN(C(C(c2c(C)noc2C)CC)=O)CC)ccc2nn[nH]c2c1 N1(C(=O)NCC2CCN(CCC)C2)CC2(CCC(C)(C)O2)C1 C(=O)(C1CNC(=O)c2ccccc21)NCC1CCC(NC(C2C(=C)CC2)=O)CC1 CCC(CNC(=O)C(C(C)C)NC(=O)Cn1ccnc1)C(C)(F)F c1(OC)ccc(Cl)c(C)c1C(=O)NC1CC(CNC(C2(N(C)C)CCC2)=O)C1 c1(C(=O)NCC2C(C)CN(C(c3cscn3)=O)CC2)ccc(C#CC2CC2)cc1 C1(NC(CC(=O)NCC2CC2)=O)CCOC12CCN(C(=O)C=CBr)CC2 c1(C(N2CC(N(C(c3c(CC)cc[nH]3)=O)C)C(O)C2)=O)cn2cccc(F)c2n1 C1(NC(C(CC)(F)F)=O)CCN(C(=O)C(C)C(=O)OC(C)(C)C)C12CC2 C1(CNC(C2(O)CCN(c3ccccc3)C2=O)=O)CC1C1CCCCC1 N12CCCCC3(C1)CN(C3)C2=O.CC(C(C)C(=O)OC(C)(C)C)C(C)(C)C C1(NC(CC(=O)NCC)=O)CCCN(C(=O)Cc2cncn2C2CC2)C1C c1(C(N(C)CC2N(C(=O)COCCF)CCC2(C)C)=O)ccnc2c1ncn2C C1(NC(c2c(CC)[nH]nc2Cl)=O)CCCCCN(C(C2CC(C)(CC)C2)=O)C1 C1(NC(C2C=CCC2)=O)CCC2(CC1)CCN(C(=O)COCC(F)(F)F)C2 C(=O)(C1=CCC(NC(=O)Cc2csc(C)n2)C1)NC(CN(CC)CC)C C(CCC(=O)NCCCC1CN(C(=O)C(c2cnn(C)c2)O)C1)OC(C)(C)C c1(C(N(C2CCCC(CNC(CN(C)C)=O)C2)C)=O)cncc2c1CCC2 Cc1c(C(=O)NC2CCN(c3nccc(C(C)(C)C)n3)C(C)C2)cncc1Cl C1(CNC(C(CC)(C)C)=O)CC2(CCC2)CN1C(=O)CC1CCC(=O)OC1 c1(C2(CCC(=O)NCCCCn3cc(Cl)cn3)CC2)ncccn1 c1(C(C(=O)NCCC2(NC(=O)CCCc3cncs3)CC2)SC)cccc(Cl)c1 Cc1cc(OC(C)C(=O)NC2(NCC(=O)O)CC2)cc(C)c1.c12ccc(cc1)o2 C(CCCCCNC(C1C2CCCCC12)=O)N(C(c1cn(CC=C)nn1)=O)C C1(C(=O)NC2(CNC(C3CC(C)(O)C3)=O)CC(OC)C2)CC2CCC1C2 C1(SC(C)C(=O)Nc2ccc(F)c(F)c2F)CCC2COCCC2C1 CC(C)C(C(C)NC(C1CC(N(C)C)C1)=O)NC(c1cncc(O)c1)=O c1(C(=O)NCCCN(C(=O)C(C)(F)C(=O)OC)CC)c(F)ccc(C)c1Cl C#CC1CN(C(C2CCCN2CC)=O)CCN1C(=O)C=CCN(CC)CC c1(C(N2CCN(C(C=C3CCC(C)(C)CC3)=O)CC2)=O)noc2c1CCCCC2 c12cnc(nc1O)CNC2=O.CCC(F)(F)C(=O)N1CCC(O)(C2CCC2)C1 C(=O)(C(CO)C(C)(C)C)NC1CN(C(C(CC(=C)C)OC)=O)CC1O C1(OC)CCCC1N=c1[nH]c(=NCc2c(Cl)cccc2Br)[nH]c2c1CCC2 c1(C(=O)NC2CCCN(C(C3(CO)CCNC3=O)=O)CC2)cc2ccccc2o1 N1(C(CC2(C=C)CCC2)=O)CCC(C2CN(C(c3ccccc3CO)=O)C2)C1 C(CC(C(C)(C)C)NC(c1cnc(O)o1)=O)N(C(=O)CC1(O)CCCCC1)C c1(C(N2CC(NC(c3c(C)scn3)=O)C(C(F)F)C2)=O)coc2c(F)cccc12 c1(OCC)cccc(C(N2CCN(Cc3csc(C)n3)CC2)C(=O)NC2CC2)c1 C12(NC(C(CC)OC3CCCCC3)=O)CC(CNC(C3CC3(F)F)=O)(C1)OC2C C(C)(CCCCNC(=O)CN1CCN(C2CC2)C1=O)NC(c1cc(OC)no1)=O S(=O)(=O)(c1cncc(C(=O)OC)c1)N1C(C)CCC(C(=O)OC)C1 c1(C(CC)N(C)C(C2CCN(C(=O)C(C)Cn3cccn3)C2)=O)ccccn1 Cn1cc(C(N2CCN(C(=O)C#CC3CCCCC3)CC2)=O)c2cccc(Cl)c12 N1(C(=O)NCc2ccc(-n3cc(-c4scc(C)c4)nn3)cc2)CCN(CC)C2CC12 C1(C(=O)NCC2C(C)(C)CCCO2)CCCN1NC(=O)C(=O)NCCN N1(C(c2cnc(CCCC)s2)=O)CCCC2(NC(c3ccncc3)=O)CCCC12 N1(CCN2CCC(CN(C(=O)C(O)CN3CCCC3)CC)C2)CCCC1=O c1(C(=O)NC2(CNC(=O)C(F)n3cccn3)CCC2)ccc2c(c1)C(=O)CCS2 c1(C(N2C3CN(C(C(CCSC)OC)=O)C(C3)C2)=O)ccc2c(n1)CCC2 C(N=c1[nH]c2c(c(=NCC(C)CO)[nH]1)CCC2)c1c(C)nccc1 Cc1c(C(=O)NC2CC(NC(C3(COC(F)(F)F)CC3)=O)C2)cc(C2CC2)n1C c1(Cc2cc(C)ncc2)ccc(C=CC(C)C)cc1Cl CCC(CN1CCCC1)N=c1[nH]c(=N)[nH]c(=NC(C)c2cc(OC)cc(F)c2)[nH]1 N1(C(Cn2ccc(C)n2)=O)CCC(C(=O)NCC2CCC2(F)F)C1C CC1CN(C)C(C)CN1C(=O)C1=CCN(C(=O)CCC2CCCN2C)C1 c1(C(=O)NC(CNC(c2[nH]cc(C)c2)=O)C)ccc(C)c2c1NCCC2 C1(C(N2C(COCC#C)CCC2)=O)(NC(c2n[nH]cc2Cl)=O)CCCC1C N1(C(c2cn(CC)nn2)C(=O)NCCCC)CC(C2(O)CCC2)C12CCC2 CC1(C(N2CC(C(N)=O)(CNC(c3cccnc3)=O)C2)=O)CCCS1 c1(OC)cnc(C(=O)NC2CN(C(=O)CCCn3cccc3)CCC2O)c(F)c1 N1(CC)CC(C(=O)NCCN(C(=O)C(c2nc(C)cs2)C)C(C)C)CC1=O c1(C(N(C)P(C)(C)=O)CCNc2ccccc2)ccc(Cl)cc1F c1(C(=O)NC2CCN(C(CCCNC(=O)OC)=O)C23CC3)cnc2nccn2c1 c1(NCc2c(C)ocn2)ncnc(NC2(c3ccccc3)CC2C)c1C C1(C(=O)NOCC(F)F)(C(N(C)Cc2csnc2Cl)=O)CC1(C)C C1(CC(=O)OC)CCCN(c2nnc(Cc3ccc(Cl)cc3)n2C)C1 n1(CCC)ncnc1CNC(=O)C=CC(C)NC(C1CC2CC2C1)=O c1(CC(=O)NC2CN(C(C=CCOC)=O)CC(F)(F)C2)ccc2c(c1)CCCO2 CCCCCCC(C)C(=O)N1CCC2CCC(C1)N2C(=O)C(C)CCO C1(C(NOCC=CC)=O)CCCN1C(c1cnc(C2CC2=C(C)C)o1)=O CC1CCSCCN1C(=O)C(Cc1cnc[nH]1)NC(=O)C(F)(F)C(F)F N1(C(CC2CCN(C(CCCCCC)=O)C2)=O)CCC2(COC(=O)N2)C1 C(=O)(C#CC(C)(C)C)NCc1c(NC(=O)NCCCOC)c[nH]n1 C1(NC(c2c(Cl)cc(C)c(C)c2)=O)CCN(C(C2OCCCO2)=O)C12CCCC2 CCC(C)CC(CO)NC(=O)CCC1(NC(=O)C(=O)NCC(F)F)CCCC1 Cc1cc(-c2ccccc2CO)ccc1-n1c(C)cnc1N1CCNC(=O)C1 c1(C(=O)NC2C=CCN(C(C(C(=O)OCC)OC)=O)C2)cccc(C)c1Br c1(CCCC)ccc(CC(=O)NCCC(C)NC(=O)C(C)(C)COCC)cc1 N1(C(c2occ(C(C)=O)c2)=O)CCC(F)(CNC(C2CCCC(C)CC2)=O)CC1 C(=O)(C(O)C(C)(C)C)NCCCNCC(=O)N(C(C(CC)C#N)=O)C1CC1 c1(-c2n(CC3CCN(C)C3)ccn2)ccc(-c2cnn(C)c2CN)cc1F C(c1ccc2c(c1)CCO2)=CC(=O)NC1CC(F)(F)CC1Cc1ccco1 N1(C(N2CC(NC(CC=C=C)=O)C2)=O)CCC(O)C(F)(F)C1 C12(C(=O)NC3(CNC(=O)CCCCO)CCCCC3)C3CCC(CC13)C2(F)F C(=O)(CCC(CC)OC)N1CC(CCC)C(C(=O)NCC(CC(C)C)N(C)C)C1 CC1(C)CCC(CNC(=O)C=Cc2ccc(F)cc2)N(C(C2CC2)C2CC2)C1 c1(C(=O)NC(CNC(CC2C(C)CCC2)=O)C)c(F)c(F)cc(F)c1F c1(NCC(C)S(N)(=O)=O)cc(S(=O)(=O)NCCSC2CCCCC2)ccc1C#N C(c1cc(F)c(F)c(F)c1)=CC(=O)Nc1ccc(NC(=O)C2CC2)cc1.C1C(=O)N1 c1(C(=O)OCC)ccc(C(=O)NCCCCC(C)NC(=O)CN(C)CC)nc1 C#CCCC(O)C(=O)N1CCOC(CCNC(=O)CCNC(=O)C(C)(C)C)C1 C#CC1(C(N2CCC(C(=O)NCc3cn(C)nc3OC)CC2)=O)CCCC1 C(=O)(C(C)CC(C)C)NCCONC(=O)C(C)OCCNC(C)=O.C#CCO c1(C(=O)NCCCN(C(C2CC(=O)NC2)=O)C2CC2)cccc(-c2nccs2)c1 c1(NC(CCCNC(C2(COCC)CC2)=O)C)ncc2c(ncn2C)n1 N1(C(CC(C(C)=O)(C)C)=O)C2CCC1CN(C(=O)C(C)n1ccnn1)CC2 C1(C(N(CCSC)CC)=O)CC2(CCC2)CN1C(C1C=CCCC1)=O c1(NC(c2ccc(OCC)cc2)=O)cc2c(cc1OC)Sc1ccccc1S2 Cc1cnn(C(C)C(=O)NCC(=O)NCC(=O)N(CCc2cn[nH]c2)C2CC2)c1 N1(C(C(=O)NCC)=O)CCC2CCN(C(=O)C=Cc3scnc3C)CC12 C12(NC(CCC(=O)NCCC)=O)CC(CNC(c3ccc(C)cn3)=O)(C1)OC2C c1(C(N2CCC(CCNC(C(C)n3ccnc3)=O)CC2)=O)cc2n(n1)CCCN2 C(C(C)C(=O)N(C(C)CC(=O)OC)C)NC(CC1(OCC)CCC1)=O CCCC(CCNC(=O)C(C)(CNC(c1c[n+]([O-])c(C)cn1)=O)CC)CCC C1(CCCC(=O)NC(C)CC2CN(C(=O)C(F)=CCCF)C2)CCCC(=O)N1 C1(O)(CC(=O)NC(CCN(C(C2(C#C)CC2)=O)C)C)CCCC1 n1(CCC(=O)NC2C(C)N(C(C3CC(C)(F)C3)=O)CC2)sc2ccccc2c1=O C1(OCCNC(C=CCOC)=O)CCN(C(C2CC2(C)C(F)(F)F)=O)CC1 c1(C(CCC)C)nc(-c2cncc(CO)c2)n(C2CC(C(=O)N(C)C)C2)n1 N1(C(c2cc(C)n(C)c2)=O)CCCCCC1CNC(=O)Cc1cnnn1C c1(CC)cccc2sc(NC(=O)NCCc3ncc(-c4ccc(F)cc4)o3)nc12 C1(NC(C(CSC)O)=O)CCN(C(c2cc(C)n(C(F)F)n2)=O)CC(O)C1 CC(C(F)(F)C(F)(F)F)=CC(=O)C(C=CC(=O)NCCCOCCNC)CC C1(C(=O)NC2C(NC(CCOC)=O)C2)CCS(=O)(=O)N1C N1(C(C(=O)NC(C)C)=O)CCN(C)CC1C(=O)N(C(C)CC(N)=O)C N#Cc1ccc(NC(C2CC(NCc3ccc(I)cc3O)C2)=O)c(Br)c1 N1(C(CN(c2ccccc2)C)=O)CCC2CCC(C1)N2C(=O)CCCC1CCC1 C1(CNC(CN2CC(C(=O)OCC)C2)=O)CC(C)N(C(c2ccnnc2)=O)C1 Cc1nc(NC(C2(F)CCC2)=O)sc1C(=O)Nc1cc(-c2ccccc2)ncn1 Cc1ccc(N)c(C(=O)NC2CC(NC(c3cc4c[nH]nc4s3)=O)C2)c1 c1(C(=O)NCCC(C)N(C)C(C2CCC=CCCC2)=O)cnc(O)c(Cl)c1 N1(C(C2N(C)CC(O)CC2)=O)CC2CCC(C1)C(NC(c1ccc(F)o1)=O)C2 c1(OC)ccc(CC(=O)NC2CCN(C(=O)CCCCSC)CC2C)c(Cl)c1 c1(C(N(CCCNC(C2CCC(F)C2)=O)C(C)C)=O)cc2c(F)cccc2[nH]1 c1(C(=O)NCCCCNC(COc2ccc(C)cc2)=O)nn(C)c2c1CCC2 C=CC1(CC(=O)NC2CC(NC(=O)C(CC)SC)C2)CCCCC1 c1(CC)nc(C)[nH]c1C(N1CCC(C)(CNc2nccc(OCC)n2)C1)=O c1(OCC)ncc(Cl)cc1C(=O)NCC1CCCCN1C(=O)Cc1nc(=N)[nH][nH]1 N1(C(C(c2nc(C)sc2)=O)=O)CCOCC(CNC(C2(C)CC3CC3C2)=O)C1 C1(C(=O)Nc2c(C)n[nH]c2)CCC2(CCN(C(C3CCC(C)CC3)=O)CC2)C1 c1(OCC)cc(C(N2CCCN(C(c3c(OC)noc3C)=O)CC2)=O)oc(=O)c1 c1(C(=O)NC2CN(C(C3CCC(C)CC3)=O)CC23CC3)n[nH]c2c1CCSC2 CCC(C(=O)OC)C(=O)NCCN1CCN(C(=O)C(N)=O)CC1.C1(C)COC(C)C1 N1(C(CC=CC)=O)CCCN(C(=O)C(C)=CC2CC2)C(C)C1 N1(C(C2CCN(CC)C2)=O)CCOC2CN(C(C3(C#N)CCCCCC3)=O)CC12 Cn1cnc2[nH]c(C(N3C4CCC3CC(NC(=O)CCC(F)(F)F)C4)=O)cc12 C(=O)(CC(C)C(F)F)NCc1nc(C(=O)NC(CN(CCCC)C)C)c(C)o1 S(=O)(=O)(c1ccc2nc(N3CCC(C(F)F)C3)ccc2c1)N(CC#CC)C C(CCC(C)(C)NC(c1cnc(OC)s1)=O)NC(CC=C)=O c12ccccc1S2.C(C(CNC(c1scnc1C(C)C)=O)CO)NC(CC=C)=O C1(NC(C2C(CC)C2)=O)CC2CCC(C1)N2C(=O)C1=COCC1 C1(C(=O)Nc2cnn(C3CCOCC3)c2)C2CN(Cc3ccc(O)cn3)CC12 Cc1cc(N(CC(C)NC(c2ccc(F)cc2)=O)C)nc(C2CC2)n1 c1(C(N2C(CNC(c3ccc(C)cc3)=O)C3CC3C2)=O)cc2sccc2n1C c1(NCC2CC(NC(COC(C)(C)C)=O)C2)cccnc1 c1(CNC(=O)NC(C(c2ccccc2Br)OC)C)ccc(C)nc1O c1(NC(C2(C)CCN2C(=O)CCCCCBr)=O)cccc2c1CC(=O)N2 C1(NC(c2c(CC)n(CC)nc2)=O)CCN(C(=O)CC2CN(C(C)=O)C2)C(C)C1 N1(Cc2cn(CC)nn2)CCCC(NC(C2CCCCC2)=O)C1 CC1(C)CCC(CNC(=O)COC2CC2)N(C(=O)Cc2cccnc2)C1 c1(C(N2CC(NC(C(CC=CCC)C)=O)C(C)(C)C2)=O)ccc2c(c1)OCC2 Cc1ccc(NS(C)(=O)=O)c(C(=O)NC2C(C(=O)NCc3cccc(F)c3)C2)c1 C1(CNC(C2(C)CC2(Br)Br)=O)CC(NC(=O)CNC=O)CC1O C1(CNC(c2cnc(C(F)(F)F)s2)=O)CN(C(C2CC=CC2)=O)C2CC12 C1(C)(C(=O)NC2C(CNC(C3N(C)CCC3)=O)CCCC2)CC2CCC(C1)S2 c1(C(C)C2CC2)ncc2c(n1)CC1CCC2N1S(=O)(=O)C1CCN(C2CC2)C1 Cc1ccc(C(CNC(C2(F)CC=CC2)=O)NC(C2COCCO2)=O)cc1 Cc1nc(O)[nH]c1C(=O)NC1(C2CCCCN2C(=O)CC2C(C)(C)C2(C)C)CC1 C=CC(CC)C(=O)N1CCC(CN(C(=O)Cn2c(C)ccc2C)CC)CC1 C(=O)(C1=CCC2(COC2)OC1)N1CC(O)(CCNC(Cc2cccc(C)c2)=O)C1 CC1CC(n2cc(C3CCN(C(=O)C(O)CO)CC3)nn2)CC(C)C1 N1(C(c2c(C)n[nH]c2)=O)CC(NC(c2cccc(C(F)(F)F)c2C)=O)C(C)(C)C1 c1(C(=O)NCC2CC(CNC(c3ccccn3)=O)CO2)cncc(Cl)c1Cl c1(C(=O)NCCC(=O)NCC(C)N(C(C2C(C=C)CC2)=O)C)ccc(F)cc1 N1(C(c2cn(C)nc2)=O)CCN(Cc2conc2C(F)(F)F)CC1 c1(NC(C2CC2NC(C2C(NC(CC3(C)CC3)=O)C2)=O)=O)cccc(CO)c1 c1(C(N(C2CCCCC2NC(C2CC2F)=O)C)=O)cnnc(-c2ccccc2)c1 c1(NC(=O)NC(c2ccccc2OC)C(=O)OC)ccc(SC)c([N+](=O)[O-])c1 C1(CC)(NC(=O)Cc2occc2C)CCN(C(C2(C(F)F)CCOCC2)=O)CC1 C=C(C)CCCNC(C1CCN(C(=O)C(C)NC(=O)C2CC2)C1)=O N1(C(=O)OC(C)(C)C)CCCC(C2CCN(c3c(C#N)ccc(Br)c3F)C2)C1 c1(CNC(=O)NC2CC2N2CC(C(C)(C)C)C2)cccc(C(=O)OCCO)c1 C1(NC(Cn2c(C)ccn2)=O)CN(C(=O)C2=COCCO2)CC1N=[N+]=[N-] c1(-c2[nH]cc(C(N(CC(C)NC(c3ccoc3Cl)=O)C)=O)n2)cccc(Cl)c1 N1(C(CC2(C)CCOC2)=O)CC2CC(C(=O)NCCCCCCC3CC3)C(C2)C1 c1(CNC(c2cc(-c3ccccc3)on2)C)onc(C(=O)O)c1Br C1(CNC(C(C)=CC)=O)C(C2CC2)CCN1C(C1CC(c2cnc(O)[nH]2)C1)=O c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CC2)nc2sc(C)cn2c1C Cc1cncc(CC(N2CCN(C(c3c(C)[nH][nH]c3=N)=O)CC2)=O)c1 c1(C(=O)NCC(C2CCN(C(=O)C=CBr)CC2)C)ccc2c(c1)nnn2C Cc1ccc(N)c(C(=O)N(CCCCNC(c2cnn3ncccc23)=O)C)c1F N(C(=NCN1CCCC1=O)NN1C(N)CC1)Cc1scc(C)n1.CC(C)(C)C c1(C(N2CC(NC(=O)CCNC(c3ccco3)=O)C2)=O)ccc2ccnn2c1.NCO C=C1CC2CC1CN2C(C1(CNC(=O)CC2(C)CC(F)(F)C2)CCCO1)=O C12(C(C)C)CC(C(=O)NCC3CCN3C(c3ccc(C(C)(C)C)[nH]3)=O)(C1)C2 c1(C(=O)NCC(CN(C(CC(CCC)O)=O)C)O)c(F)ccc(Br)c1C Cc1ccc(C(CNC(=O)C(C)O)NC(=O)C(C)(C)C2CCC2)cc1 CCC(C)C(CC(=O)NCc1ccnc(O)c1)NC(C1CC(=O)CS1)=O c1(CC(C(=O)NC(CC)C)NC(c2ns[nH]c2=O)=O)ccc(Br)c(OC)c1 c1(C(=O)NC2(CO)CCN(C(CC(CC)C)=O)C2)ncc(C#N)cc1Cl C1(C(=O)NC(CC)C)C=CCN(C(c2cc(Cl)cn2C)=O)C1 Cc1ccc2c(c1)CCC(C(=O)NC(C)CNC(C13CC(F)(C1)C3)=O)O2 N1(C(C(C)(O)C2CC2)=O)CCN(C(=O)Cc2cccc(F)c2F)CC1CF C(C(CC(C)C)C(=O)N(CC)Cc1ccccc1)NC(COCCC#C)=O N1(C(Cc2c(C)n(C)nc2)=O)CCCCC12CN(C(C1CCOC1C(C)C)=O)C2 C1(CNC(C(C(C)C)NC(c2cncc(C)c2)=O)=O)Cc2nccn2C1 C(CCCCCC(=O)NC(C)(C)CCF)NC(c1cc(C(C)C)[nH]n1)=O CC1(C(=O)NC2CC(NC(C3COCCN3C3CCCC3)=O)C2)CS(=O)(=O)C1 c1(CNC(c2c(CNC(C(CC)NC(N)=O)=O)noc2)=O)ccccc1F C(=O)(C1=CC2(CN(CC3CCCN(C)C3)C2)OC1)N1CC(C(C)(C)C)OCC1 C1(O)(CNC(=O)Cc2ccns2)CCCN(C(c2ccc(C(F)(F)F)cn2)=O)C1 CN1CCC(C(=O)NCC(c2ccccc2)CNC(c2cc(CO)on2)=O)C1 Cc1ncc(CC(=O)NCC2C(C)CCN2C(=O)CC2(C)CC2)c(O)n1 C1(OC)(CNC(c2cc(F)c[nH]2)=O)CN(C(c2ccsc2C(=O)OC)=O)C1 CC1CN(C(C2CCN(C)CC2)=O)CC1CNC(c1ccc(-c2cccs2)o1)=O N1(C(c2c(C)[nH][nH]c2=N)=O)CCC2(C1)CN(C(c1ncsc1C1CC1)=O)C2 N1(C(CCC(=C)C)=O)CCC2(CCC2NC(=O)CC2=CCCCC2)CC1 S(=O)(=O)(c1ccc(NCC23CC(CN2C)C3)c(C#N)c1)N1CC(C)OCC1C c1(CC(=O)NC(C2CCN(C(c3cncc(CC)c3)=O)C2)C)cc(C)ccc1C c1(C(=O)NC2CC(CNC(C3(C)CCCC3(F)F)=O)C2)ccc2c(c1)CNC2=O S(=O)(=O)(c1ccccn1)N1C(CNC(c2cc(OCC)c(O)cc2)=O)C=CC1 Cc1cc(C)c(NC(=O)C(N2CC(C(=O)OC)CC(C)C2)C2CCC=CO2)c(C)c1 CCC(C)(C)OC1CC(NC(=O)CONCN2CCC2=O)C1 c1(C(N2CC(SC)C(NC(=O)CC3=NNC(=O)C3)C2)=O)c(Cl)ccc(Cl)c1O C1(O)(CNC(C2CCN(C(C)C)C2)=O)CCN(C(=O)C(F)=C2CCC2)C1 c1(CS(C)(=O)=O)ccc(NC(C2CC3CC3N2Cc2ccc[nH]2)=O)cc1 c1(CC(=O)NC(CNC(c2c(OCC)ccc(C)n2)=O)C)cn2c(C)csc2n1 C1(C(N(C)CC2(O)CN(C(=O)Cc3ccnn3C)C2)=O)CCCC2(CCC2)O1 c1(C(=O)NCC=CCNC(=O)NC)ccccc1CNC(=O)C=Cc1ncc[nH]1 C1(NC(C(CCF)NC(c2c(CC)ncs2)=O)=O)CN(C)CCN(C)C1 CC#CCC(C(=O)NCC1CC[Si](C)(C)C1)NC(=O)C(O)Cn1cncn1 C1(C(N2CC(COC)C2)=O)C2CC3C(C2NC(C2(C(C)(F)F)CC2)=O)C13 C1(CC(N2CC(C)(C(=O)NCC(C(C)C)O)C2)=O)CCCOCC1 Cc1cc(Cl)c(C(=O)NCC(C)(C)CNC(C2(C(O)C(F)(F)F)CC2)=O)cc1F Cn1nc(C(=O)NCCC(O)CNC(C2(F)CCCOC2)=O)cc1Cl N=c1nc(O)cc(C2CC2)[nH]1.C1CCCNC(=O)N1 N1(C(c2occ(C)c2C)=O)C(CNC(c2coc(Cl)n2)=O)CC2CCCC12 N1(C(Cn2nc(C)oc2=O)=O)CC23CCCCC2(C1)CN(C(C1CC1(Cl)Cl)=O)C3 N#Cc1cccc(C(C(F)(F)F)NC(c2ccccc2Cl)=O)n1 c1(OC(CC)C)ccccc1C=CC(N1CC=CC(NC(C2CC2F)=O)C1)=O C1(C(=O)NCC2N(C(CC3CCC(OC)CC3)=O)CCCC2)Cc2cscc2C1 C1(NC(C(C)OCCC#C)=O)CC(C)(CNC(c2ccccn2)=O)C1 C1(C(C)C)CN(C(=O)C(C)C)CCC1NC(=O)C(C(C)C)N1CCCCC1 CS(=O)(=O)c1coc(C(N2CC(NC(=O)CCCCCF)C(C(F)F)C2)=O)c1 C=CCCC(C(=O)N1CCN(C(C2CCC(=O)O2)=O)CC1CC(F)F)OC C1(CNC(C(C2CCC2)OC)=O)CN(c2ncc(I)cn2)CCCO1 C1(CC)CN(C(=O)CCC2(C)CC2)CCN1C(=O)Cc1nnc(C)o1 CC(C(=O)NC1CN(C(C2(c3ccncc3)CC2)=O)CC1C(F)F)C(F)F Cc1nn(C)c(Cl)c1C=CC(=O)NCC1CCN(C(c2ccccn2)=O)C1(C)C c1(C(=O)NCCCOCCNC(C(C)(C)C2CC2)=O)ccc2cccnn12 N1(C(CC2(C)CCN2C(C2CCCC(CO)CC2)=O)=O)CCOC2(CC2)C1 N1(CCCN(C)C)CCCC(C(=O)N(C(C)(C)C)CC2CCOCC2)CC1 c1(NCc2ccc(C(N3CCC3C(=O)OC)=O)cc2F)cnc2cccnn12 N1(C(C(CC#C)O)=O)CCCC2(CCCCN2NC)C1.C(C)(C)(C)OC=O C1(C(=O)OCC)CCCCN1CCOC(C)(C)C.C1(C)(C)C(=O)N1 N1(C(c2c(CNC(C(CCC)OCC)=O)nnn2C)=O)CCC(C)(CC)CC1 Cc1cccc(C)c1-n1nnnc1C(C)(CCI)NCCc1cccc(I)c1 C1(C(=O)OC(C)(C)C)CCCC(C(N(CCNC(C)=O)C(C)C2CC2)=O)C1 c1(C(N2CCN(C(CC(=O)OC(C)(C)C)C)CC2)=O)cc(C(=O)OC)nn1C C1(C(=O)OC)CC(F)(F)CC1NC1CCCN(C(=O)CC23COC(C)(C2)C3)C1 CC(CN(C)C(c1coc(C2CC2)n1)=O)C(=O)N1CCC(CSC)C1 C=Cn1ncc(C(N2C(C(N3CC4CC3(C(N)=O)C4)=O)CCC23CC3)=O)c1N Cc1ccc(CC(=O)NCC(C)CNC(=O)C(C(C)C)N2CCCCC2)c(C)c1 c1(C(=O)OCC)cc(-c2csc(NCC3CCS(=O)(=O)C3)c2)ccc1F C1(S(C)(=O)=O)(C(=O)NC(CCCNC(CC(C)C)=O)C)CCCCC1 C12(NC(C(F)=CCC)=O)CCCC1CN(C(=O)Cc1c[nH]c3ccccc13)C2 C1(O)(CNC(CCC)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC1 C1(C(N2C(C(C)NC(c3c(OCC)scc3)=O)CCC2)=O)CCCC(F)(F)C1 C1(CC)CCN(C(=O)COCCCC)C(C(N2CCC=C(Cl)C2)=O)C1 c1(NC(C2OCCN(Cc3scc(C)c3)C2)=O)ccc(C(N)=O)c(F)c1 N1(C(C(COC)(F)F)=O)CCC(CO)(CNC(=O)CCc2nncs2)CC1 c1(-n2c(C(C)P(C)(C)=O)nc(C(CCC)C)n2)ccc(S(N)(=O)=O)cc1 c1(C(=O)NC(CC)CNC(C2(F)CCOC2)=O)cc(C2CC2)nc(O)c1 N#Cc1c[nH]c(=NC(=O)c2ccc(NCc3ccncc3[N+](=O)[O-])nc2)cc1F C1(OC)CN(C(c2cncs2)=O)C(C)(CNC(=O)CC#N)C1 CN1CCC2CCN(C(=O)NC3CN(Cc4ccccc4)CCO3)C2C1 C1(O)(C(C)C)CCC(NC(c2cnn(C3CC3)c2Cl)=O)C1 C(C(=O)N1CCCC(CNC(=O)Cn2ccc(O)nc2=O)C1)(C(C)C)OC C(C(CC(C)C)C(=O)NC1(CO)CCCCC1C)NC(Cc1ccc(C)o1)=O C1(CC)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C(=O)C(CO)c1ccccc1 N1(C(CC2OCC(C)(C)C2)=O)CCC(NC(c2ccnc(O)c2)=O)C(O)C1 C(C)(C(=O)NCC1(F)CC(CNC(c2cc(C)cs2)=O)C1)(C(C)C)OC C(C)(C(=O)N(CCC(=O)OC)CCOC)NCCN(C1CC1)C(C)C C1(CNC(C(COC)C)=O)CN(C(c2ccsc2C#N)=O)CC12CCOCC2 C1(C(N2CC(COC)(NC(c3nccc(Cl)c3C)=O)C2)=O)CN2CCCC2CO1 CCC(CC)C(C(=O)NCC(F)F)N(CC(N1CCOCC1)C1CCCO1)C c1(C(=O)NC(CNC(C(CCCOC)C)=O)(C)C2CCC2)ccc2[nH]ccc2c1 C=CC1COCCN1C(C1CCC(NC(c2ccc(C)n2C)=O)C1)=O CCC(C)C(O)C(=O)NCCSCc1cn(-c2ccc(C(=O)O)cc2)nn1 Cc1cc(C(=O)NCC(C)CNC(=O)Cc2cncnc2O)c(Br)cc1F c1ccccc1F.C12CCCC1C(=O)NCC(=O)NC2.n1(C)cc(CO)nn1 Cc1cnc(C=CC(=O)NC2CCCC2NC(=O)COC2CCC2)[nH]1 N1(C(c2c(C)cns2)=O)CC(C(F)(F)F)C(CNC(C2CCCCC2)=O)C1 C1(NC(c2ccc(CC)nc2)=O)CC2CC(NC(=O)CCN3CCCCC3)CC12 C(CCC(C(=O)N(c1csnc1OCC)C)NC(c1cnn(C2CC2)c1)=O)OC CCC(CC(=O)NC(C12CCC(CC1)C2)CNC(=O)CNC(=O)CO)C1CCC1 N1(C(c2cc(CC)no2)=O)CC(CCNC(=O)CCc2ccccn2)C(C)C1 C(CNC(=O)CCC1CCCCCC1)(CC(F)(F)F)NC(CN(C)C(N)=O)=O CC(CCNC(=O)CC1(C)CCCO1)CCNC(c1coc(Cl)n1)=O N1(C(CSc2n(C)cnn2)=O)CCC(NC(c2ccon2)=O)C(F)C1 N1(C(CC2CC(OCC)C2)=O)CCC(N(C(=O)CCOC2CCOC2)C)CC1 CCC(C)N=c1[nH]c2ccc(C(=O)NC3CC(NC(=O)C(C)C(C)(F)F)C3)cc2o1 c1(OCC)cc(C(=O)NC2CCC(CCNC(c3cc(CC4CC4)n[nH]3)=O)C2)on1.SC C1(COCC(F)(F)F)CCCN(c2nnc(C3CC3)n2CC2=NOC(C)C2)C1C C1(C(C(=O)NC(C)CCC2CCCO2)N)(C(=O)N(C)C)CCOCC1 c1(C(N2CC(CNC(c3ccc[nH]3)=O)OCCC2)=O)ccc2ncccc2c1F C1(CN(c2ccc(Cl)cc2)CC(C)(C)C)COCC(C)(C)O1 C1(NC(CC(C)N(C)C)=O)CCCCC1NC(=O)Cc1cnco1 C=C(Cl)CC(C(=O)NCC1(COC)CCCC1)NC(=O)C(C)CO N1(C(CC(=C)C)=O)C2CCCC1CN(C(c1cccnc1NC(C)C)=O)C2 C1(N(C)C(c2cccnc2O)=O)CCCN(C(c2cnc(O)s2)=O)CC1 N=c1[nH]c(Cl)c(Cl)cc1C(=O)NC12CCN(C(c3csc(O)n3)=O)CCC1C2 C1(C(=O)NC(C2N(C(C3(C=C)CC3)=O)CCC2)C)CCCCNC1=O c1(C(=O)NCC(C)(CC)NC(c2ccc(CC)c(C)c2)=O)nc2c(s1)COCC2 N1(C(c2ccncn2)=O)CC2(CC(C(N3CCC4CC34)=O)CO2)C1 C1(C(=O)NC(C2CCN(C(C(CC=C)(F)F)=O)C2)(C)C)CCc2ncncc2C1 N1(C(CCN(C(CCC)C)C)=O)CCC2C(C3SCCN3C(=O)C(CC)OC)C2C1 C1(NCCC2CCN(C(C(N)=O)=O)CC2)CCn2c(O)nnc2C1 CC1CCCC(C)N1C(C1CCCN(Cc2csc(C(F)(F)F)n2)C1)=O N1(C(c2c(CC)n(C)cc2)=O)CC2CC(C1)N2C(C1(CC2CC2)CCC1)=O c1(CCC(=O)NCC(C)N(C(C2CC(CC(F)F)C2)=O)CC)nnc(N)[nH]1 CCCCCCCCC(C)CC(=O)NC(C)C(C)NC(c1csc(Cl)c1)=O O=C(C1=CCOC1)NN(CC(F)(F)F)CCc1ccccc1.C12CCC13CC23 C1(NC(=O)CC(O)CC2CN(C(C3(C(=O)OC)CC3)=O)C2)CCC(SC)CC1 N1(C(c2c(OC)cccc2)=O)C2CCC1C(CNC(c1cc(C)nc(O)n1)=O)C2 Cc1nn2ccccc2c1C(N1CC(CCNC(=O)C(C)CSC(F)(F)F)C1)=O c1(OC)ccc2c(n1)NC(C(N1CCC(C(C)NC(c3nocc3C)=O)C1)=O)C2 C(=O)(C(CC(=C)Cl)NC(c1ccn(C(C)C)n1)=O)N(CC#C)C(C)C C(CC(C)(C)CC(=O)NCC=CC(N1CC1CC1CCCC1)=O)OC C1(C(=O)NC2CCC(N(C(=O)CCCF)C)CC2)CCCCN1S(N)(=O)=O C(C(C)(C)CC(=O)N(CCCOCCCNC(=O)C(C)n1ccnc1)C)OCC C#Cc1ccc(C(N2CC(O)(C(C)NC(c3cnn(CCF)c3)=O)C2)=O)cc1F C1(C(N(C)CCN(C)C)=O)CN(C(C2CC(N(C)C)C2)=O)CCO1 C1(C(=O)NCC)CC2CCC1N(C(=O)CCc1ccccc1C)C2 c1(CC)ccc(CC(=O)N(CC(O)CN(C(=O)C(C(C)OC)N(C)C)C)C)cc1 C1(C(=O)NC2(C)CC(NC(c3ccncc3Cl)=O)C2)CCc2nc[nH]c2C1 C(=O)(CCCC(C)(C)C)NC12C(CN(C(C(C)(c3ccccc3)N(C)C)=O)C1)C2 N1(C(CC(C)n2cccn2)=O)CCC2(CCCN(C(=O)CCC#N)C2)C1 N(C(=NCCC(=O)N1CCC1)N1CCC(CS(C)(=O)=O)C1)C(C)C c1(C(=O)NCC23C(CN(C(CC(C)C)=O)C2)C3)cc([N+](=O)[O-])c(Cl)cc1F C(=O)(C1=NOC(CNC(c2cccc[n+]2[O-])=O)C1)N(CC(C)(C)O)CC N1(C(C(C=C)OC)=O)CCC12CN(C(=O)CC1CCCN1C)C2 CCCS(=O)(=O)CC(=O)N1CC2CCOC2(CNC(C2CC2(C)C)=O)C1 C(c1ccncc1)=C(C)C(=O)NCC1CN(C(c2oncc2C)=O)C2CC12 N1(C(C2CCN(C(=O)NC)CC2)=O)CC(NC(C2(CF)CC2)=O)CC(C)(C)C1 C[Si](C)(C)c1cccc(-c2ccc(C(=O)Nc3cc4sccn4c3)c(F)c2)c1 c1(CC(=O)NCC2CCC(NC(=O)C(O)CC3CC3)C2)ccc(F)c(Cl)c1F c1(C(=O)Nc2c(OCc3cn(C)nc3)ccc(F)c2)cc2ccc(O)nc2s1 O=CC1=CCCCCC1.C1(c2cn(CC(=O)O)nn2)CC12C(=O)Nc1ccccc12 c1(NC(=O)NC(CC(=O)OC)C(C)(C)C)cc(F)cc([N+](=O)[O-])c1 c1(NCC2(CCNC(c3ccc4ncsc4c3)=O)CC2)nc2cc(Br)cnc2s1 Cc1ccc(CCC(=O)N(C)CCN(C(=O)COCC(F)F)C)cc1Cl C1(NC(c2ccc(CC)cc2)=O)CCN(C(c2csc(CC)n2)=O)CC1O CCC(C(F)(F)F)NC(CC(C)C)c1nnnn1C1CCOCC1 c1(NC(=O)NCCN(CC(CC)(C)c2cnccn2)C)ccc(F)c(OC)c1 C(C1=CCCN(C(=O)C(=Cc2ccccc2)C)C1)NC(CN(C(C)=O)C)=O C1(COc2[nH]cc(CC)n2)CN(C(=O)CCCCn2ccnn2)CCO1 c1(C(N2CCN(CCO)CC2)=O)cnc(OCCC(F)(F)F)cn1 Cc1cnccc1CN(C)C(c1ccc(CNC(=O)CC2CC2C2CC2)o1)=O C1(C(=O)NC(CNC(CC(C)C)=O)(C)C)COc2ccc(C(=O)O)cc2C1 c1(C(N2CC3C(C(=O)NCC(CC)CC)(CC3)C2)=O)ccnc2ccccc12 C1(CC)CCC(C)N(C(C23CC(C(C)(C)C)(C2)C3)=O)C1 C1(NC(=O)CCSC(F)(F)F)CN(C(C2CC23CCOC3)=O)CC12CCC2 c1(OC)ccc2cc(NC(=O)NC(C)Cc3cnccn3)ccc2c1 C=CC(C)(O)C(=O)NCCC1(CNC(C2CC(COC)C2)=O)CC1 C(c1cccc(O)c1)=CC(=O)NC1(CCNC(=O)CC2(O)CCCOC2)CC1 C1(CC)(NC(=O)C=CCOCCOC)CCN(C(=O)CCS(C)(=O)=O)CC1 C(=O)(C#CC1CCCO1)N1CCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 c1(C(N(C2CN(C(COC(C)=O)=O)CC2(C)C)C)=O)ccc2cncn2c1 c1(CC)noc(CCNC(C2(NC(=O)CCC3CC3(C)C)CC(COC)C2)=O)n1 c1(C(N(C2CCCC2)CCCNC(C=CCCC)=O)=O)cc(CCN(C)C)on1 N#CC1=C(C(=O)NCC2CCC(NC(c3cnc(C4CC4)nc3)=O)C2)CCC1 C1(NC(C2(C(C)(F)F)CC2)=O)COCC1n1cc(C(C2CC2)C2CC2)nn1 c1(C(=O)NC(N2CC(CO)CC(C)C2)=O)ccc2cccnc2c1 C1(CC=C)(C(=O)N(C)CCN(C)C(C2CN(C3CCC3)C2)=O)CCOC1 N1(CCNC(C2(C)CCCN2CC2CCCO2)=O)CCCCCC1=O CCC(CC(=O)N1CC=CC1(C)C(=O)NCC1(O)CC(C)(C)C1)C(C)C n1(CCOC)nc(-c2ccc(F)cc2)nc1-c1ccc(CC(C)(C)C)s1 C1(NC(C2CCC(=O)O2)=O)CC(Nc2ncc(C3CC3)cn2)CC1O N1(C(CCCC)=O)CC(CNC(=O)C(C)(O)CC)OC2(CCC2)C1 CCCN=C(NCCSC1(C)COC1)NCCc1cc(C)on1 N1(C(C(CN(C)C)N(C)C)=O)CCCC1(C)C(=O)NC(C1CCCC1)CO Cc1cc(C(=O)CCC(=O)NC2CCOCC2NC(c2cnns2)=O)c(C)s1 c1(C(=O)NCCC(C)N(C(=O)C(C)CC(F)F)C)cnc2sccn12 CCCCCCCC(=O)N1CC(O)CCC1C(=O)NCc1ccn(CCF)n1 c1(CC)cc(C(=O)NCC(C)C(N2CCOC(C)C2)=O)nn1C C=CCCCC(=O)NCC(C1CCCN1C(c1cc(-c2ccco2)c[nH]1)=O)(C)C N1(C(C23CC(C(=O)O)(C2)C3)=O)CCOCC(C(=O)Nc2cnc(C(F)F)cn2)C1 N1(C(C2C(=C)C2)=O)CCCC(CNC(c2ccc(CC(C)C)cc2)=O)C1 C1(C(=O)Nc2ccc(C#C)cn2)CC2CN(C(=O)C(F)C(C)COC)CC2C1 N1(C(CCCC#C)=O)CCN(C(c2cc(C(C)=O)c[nH]2)=O)C(COC)C1 C(=O)(C1CCCc2ncnn21)N1CCC(NC(C)=O)CC1 C1(C(C)C)(C(=O)NC(CCO)C(C)C)CCCN1C(c1csnn1)=O N1(C(C=C(C)Cl)=O)CC=C(CNC(=O)C(CN(C)C)c2ccccc2)CC1 c1(NC(C(c2sc(Br)nc2C)N(CCC)C(C)C)=O)ccc(SC(C)CC)cc1 C1(NC(c2cn(C(F)F)cn2)=O)CC2(CCN(C(=O)C=C3CCSCC3)CC2)C1 CC(C)(CC1CCC1)C(=O)NCCC1(O)CCN(C(=O)C=Cc2cc[nH]n2)C1 C1(F)(NC(=O)OC(C)(C)C)CCN(N2CCn3c(cnc3C(F)F)C2)C1 C12(CN(C(=O)CCNC(=O)Oc3nc[nH]n3)C1)C(=O)N2.C(C(O)C1(C)CC1)OC c1(NCc2cccc(CNC(c3cc(CC)n(C)n3)=O)c2)ncnc2scnc12 N1(C(c2cc(C)sc2C)=O)CCc2ccccc2C1CNC(=O)CS(C)(=O)=O C(C)(C(=O)NCC1(NC(=O)Cc2ncccc2F)CCCCC1)(C(C)C)OC Cc1nn(C)c(Cl)c1CNC1CCC(c2ccc(Br)cc2)C1 CC1CCC(S(C)(=O)=O)CN1C(c1ccc(=O)n(-c2ccc(F)cc2)c1)=O N1(C(c2c(C)nccc2)=O)CC2ON=C(CNC(C3(CC4CC4)CC3)=O)C2C1 C(c1cccc(Br)c1)=CC(=O)N(C)CC1CCC(C)CC1C(=O)OC(C)(C)C Cc1cc(C)c(C(=O)NC2(C(=O)NC(CO)CC(C)(C)C)CC(F)C2)cn1 c1(CC(=O)NCC2N(C(C(CC)C)=O)CCC2)ccccc1SC.N(CCO)C1CC1 c1(C(=O)NCC(C)NC(c2cc(C3CCOCC3)[nH]n2)=O)n[nH]c(C2CC2)c1Cl Cc1ccc(CC(N2CCC(n3cc(CNC(=O)CC4CC4C)nn3)C2)=O)cc1 c1(C(=O)NC2(CNC(CCN(C(C)=O)C)=O)CC2)cc(C2CC2)cs1 C1(CNC(C2(N)C(C)(C)C2)=O)CS(=O)(=O)CCO1 CC(C)CC(O)C(C)C(=O)N1CCOC(CC(N2CCC(O)C(C)(C)C2)=O)C1 c1(C(N2CCCC(CNC(c3c(CC)c[nH]c3)=O)C2)=O)cnc(CO)nc1C N1(C(C(CC)SC)=O)CC(C)CN(C(c2ccc3nc[nH]c3n2)=O)CC1C N1(C(CC(=O)OC)=O)CC2CC2(C(=O)N(C(C)CO)C2CC2)C1 c1(C(N2CCN(C(C(C=CC)O)=O)CC2COC)=O)cnc(O)c2ccccc12 CC1CN(CCO)CC1(c1nnnn1CCN(C)C)Nc1c(Cl)nsc1Cl c1(C(=O)NCC(N(C(C(CC)n2ccnc2)=O)C)C2CC2)cc(SC)ccc1C C(=O)(C(O)CCCC)N1C(C(=O)NC(C=C)C)COCC1 c1(C(=O)NC2CC3(C(C(=O)NCC=C(C)CN4CCCC4)C3)C2)ccc(C)nc1C C1(NC(c2ccc(C3(C)CC3)cc2)=O)CC2CC1CN(C(c1cccs1)=O)C2 N1(C(COC2(C)CCC2)=O)CCCCCCC1C(=O)NCCc1nncs1 Cc1c(N2CCC(N3CCOCC3)C2)ncnc1N1CCN2CCC2C1 c1(OC)cc(C(N2CCC=C(C(=O)NCCN(C)C)C2)=O)cc(OC)c1O C(=O)(C1=CCC2(COC2)OC1)NCC1N(C(CNS(N)(=O)=O)=O)CCC1 c1(CNC(c2cc(CC)oc2C)=O)ccc(CNC(C2(C)CC2)=O)c(F)c1 CC#CCC(C(=O)NC1CC(C(C)(C)O)C1)NC(=O)C=CC(=O)N(C)C C12(CNC(C3(CC#C)CCOCC3)=O)CCC(C1)N(C(C1CCCCS1)=O)C2 C(C)(CNC(=O)Cc1csc(C)c1)(CC(C)C)NC(C(CC)OCC)=O C1(CNC(=O)Cn2cccn2)CC2CCC1N(C(c1ccc(CO)o1)=O)C2 N1(C(C2C3CN(C(C4C(CC)CCCC4)=O)C2C3)=O)CCCC(F)CC1 C1(CC(N2C(C)CC(NC(Cn3nc(C)oc3=O)=O)C2)=O)CCC(C)(C)CO1 C1(NC(c2ccc(I)cc2F)=O)CN(C(c2cccc(F)c2F)=O)CCC1(F)F c1(NCC2(NC(C3CC4CCC3C4)=O)C(C)CCCC2)ncnc(Cl)c1[N+](=O)[O-] n1(CCC)nccc1C(=O)N(CCC(=O)N(CC(C)C(C)C)C)C1CC1 C(=O)(C(C)C(=O)N1CCCC(NC(c2n[nH]cc2OC)=O)C1)OC C1(NC(c2cccc(-n3cc(CC(C=C)O)nn3)c2)=O)CC2CC3C(C2)C13 C1(OC)CN(C(=O)CC2(N(C)C)CC2)CC1NC(=O)C(C1CCOCC1)F C1(C#N)(Cc2nc(NC(=O)NC(c3ncccc3F)C)sc2)CCOCC1 O=C1CCC(C(N2CC(OCCNC(=O)C3=NOCC3)C2)=O)CN1 C(Cc1cn[nH]c1)(C(=O)N1CCCC1CC(N)=O)NC(CC1(C)CC1)=O CC1CC(NC(=O)C=Cc2nccs2)CN(C(c2ccc(N)c(F)n2)=O)C1 Cc1ccc(O)c(C(N2C3CCC2C(C(=O)NC2(C)CCC(C)C2)C3)=O)c1 N1(C(C(CCCC)O)=O)CCC2OCCN(C(=O)C(F)(F)c3nc(C)cs3)C2C1 n1(CC)nccc1C=CC(=O)NC1(COC)CCN(C(C2(SC)CC2)=O)C1 N1(C(c2c(CC)noc2)=O)CCCC(NC(=O)C(C(C)C)NC(C2CCC2)=O)C1 N1(C(Cc2nc(C(C)OC)sc2)=O)CC(CO)C2(C1)CN(C(=O)CS(N)(=O)=O)C2 CCCCC(CC(=O)N1CCC(C)(CC)CC1)NC(c1coc(C)n1)=O C(CC(C)(C)C(=O)Nc1ccccc1F)NC(C(C)n1cccn1)=O C1(NC(=O)CC2(O)CCC2)CCN(C(=O)CCc2nc(CC3CC3)no2)CC1O N1(C(C2CN(CCC)C(=O)C2)=O)CC(CO)C2(C1)CN(C(=O)Cn1ccnn1)C2 C=CC1CCCN(C(c2cccn2CC)C(=O)Nc2ccccc2C)C1 C(=O)(C(C)CC(=O)OC)N(CCN(C(c1nn(CC)c(C)c1)=O)C(C)C)C C#CCCCC(C)C(=O)NCC(C)(C(C)C)NC(c1cc(O)nc(O)n1)=O N1(C(C(CC(C)C)(C)O)=O)CCC(CNC(=O)CC(C)(C)F)C(F)(F)CC1 Cc1cc(CC(=O)NC2CS(=O)(=O)CC2NC(c2cnc(S)n2C)=O)cc(F)c1 c1(NC2C(CNC(=O)NCC3CC3)C2)ccc([N+](=O)[O-])cc1C(F)(F)F c1(C(=O)Nc2cccc(-c3ccco3)n2)cn2cc(CO)ccc2n1 C1(NC(C(C)O)=O)CC(N=c2[nH]nc(-c3ccccc3)s2)C12CCOCC2 N1(C(C(CC)CC)=O)CCN(C(=O)Cn2ccnc2C)CC2CCCCC12 CC(c1ccccc1C)=CC(=O)NC1CC(NC(=O)CC2CCCC2O)C(O)C1 c1(NC(C(C)N(C(=O)CCF)CCNCCC#N)=O)ccc(F)cc1F Cn1ncc2cc(C(N3CCC(C(N4CC5CC5C4)=O)C(O)C3)=O)cnc12 N1(C(C2CCN(c3c(C)cnc(C)n3)CCC2CO)=O)Cc2ccccc2C1 c1(C(C)NC(CC(C)C)c2ccccn2)ccc(OC(C)(C)C)cc1 N1(C(CCCOCCC)=O)CCN(C(C2ON=C(C)C2C)=O)CC1CC1CC1 C1(C2CCN(C)CC2)(C(=O)NCCCN(C(=O)CCCC(C)(C)C)C)CC1 N1(C(C(CC=C)CC)=O)CCC(C)(C)C(C=O)C1.N1(C(=O)NC)CCC1 c1(CC)cc(C(=O)N(CC(C)NC(C2CCC=CCC2)=O)C)c2c(c1)CCO2 C(CCC(C)C)(C(=O)N1CC2(CCC(CNC(C3CSCCS3)=O)O2)C1)OC N1(C(CC(C)OC)=O)CCN(CC(=O)NC2CCCOC2)CC1 CCC(CC(=O)NCC1(OC)CCC1)OC(C)C.C12(CCCC1C)C(=O)N2 C(=O)(CCCC(=O)NC(CC1CCC1)C(=O)NC1CC1c1nn[nH]n1)OC c1(NC(C2CCCN(C(C(C)N(C)C)=O)C2)=O)ccc(C(C)(C)C)c(Cl)c1 C(CCC(=O)NCC1CC1CC(N1CCC(n2cnnn2)C1)=O)=CCC=C C1(C#CC(=O)N(CCC(C)NC(c2cc[n+]([O-])cc2)=O)C)(CC)COC1 c1(OC)ccnc(C(N2CCC(C)C2CNC(=O)C=C(C)C)=O)c1 c1(CC(N2CCCC(c3cn(CC(=O)OC)nn3)C2)=O)ccc(F)c(OC)c1 c1(C(=O)OC)cc(CNC(C(C)(C)C)Cc2ccccc2)c[nH]1 c1(C(=O)NC2C(NC(C(c3cccc(OC)c3)O)=O)C2)ccc2c(n1)CCC2 Cn1nc(CC(=O)NC2(C)CC(NC(c3csc(C#N)c3)=O)C2)cc1Cl N1(C(CCc2nc(C)sc2)=O)CCN(C(c2cn[nH]c2)=O)CC2CCCCC12 C(=O)(C(CC(=C)Cl)NC(=O)CC1C(C)(C)C1(C)C)N1CC(F)(CC)C1 C1(NC(c2scnc2Cl)=O)CC(F)CN(C(=O)CCc2cnc[nH]2)C1 C(=O)(CCCN(C)N=O)N1C(CC)CN(C(=O)C(C(C)(C)C)N(C)C)CC1 c1(OC)cc(F)c(CC(N2CC(NC(C3CCCCC3)=O)C(O)C2)=O)c(F)c1 CC1C(NC(c2cccnc2N2CCCC2)=O)CCN1C(=O)CSCC(F)F C(=O)(C1=CC(C)CC1)N(CC(c1ccccc1)NC(CCC)=O)Cc1cn[nH]c1 c1(CC(=O)NCC2CN(C(C3C(c4n(C)ncc4)OCC3)=O)C2)ccc(Cl)cn1 CC1(C)C(CO)CN1C(=O)CCOCCCNC(C1CC(F)CN1C)=O CC1CC(NC(c2cc(N3CCCC3)ccn2)=O)CN(Cc2ccccc2F)C1 CC(C(=O)NC1(CCC(=O)N(CC(Cl)Cl)C)CCC1)NC(=O)C1CC1 C1(NC(Cn2c(C)cnc2)=O)CCN(C(c2coc(Cl)n2)=O)C1(C)C N1(C(CS(CC)=O)=O)CCN(C(c2ccc(Cl)c(C)c2)=O)C(COC)C1 c1(C(=O)NC2CC(NC(C3CC(C)C3)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(c2cncc(OC)n2)=O)CC2(C1)CN(C(C1CC1c1ccc(Cl)cc1)=O)C2 CCCC(C(=O)NC(C)CCN(C)C(c1ncc(C)cn1)=O)NC(C)=O N1(C(CC(CCC)O)=O)C2CCCC1CN(C(c1c[nH]nc1C(F)F)=O)C2 C1(NC(CCCC#C)=O)CC12CCN(C(c1ccc(C)nc1OCCC)=O)C2 C1(C2CC2)(CNC(c2cc(OC)nn2C)=O)CCN(C(=O)CC(C)C2CC2)C1 c1(NC(=O)NC2CC3(CC(C)(OC)C3)C2)cc(C)c2c(O)nc(O)nc2n1 C1(CCNC(=O)CC2CCOC2)CCCN(C(=O)C=Cc2nccs2)CC1 C1(NC(c2cc(C(C)C)on2)=O)CCCCC1NC(=O)C(c1ccccc1Cl)C C(=O)(CCC(=O)NCC(C)(F)CNC(c1nnc(S)n1C)=O)N(C)C N1(C(=O)NCC2C=CCCCC2)CCN(C(c2ccccc2)=O)CC(O)C1 Oc1ncccc1CNC(=NCC1CC1)NC1CCOC(c2ccccn2)C1 C1(N(C(c2ncc(C)nc2)=O)C)CCCN(C(c2nc(C)n(C)n2)=O)CC1 N1(C(C2(CC#C)CCCCC2)=O)CCCC2(NC(c3cncc(C)c3)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)CCc2ccccc2O)C)c2c(nn1C)CCCC2 Cc1cc(C(=O)NCC(=O)NCC(=O)NCC(=O)N(C)C)nn1C CC1CCC(C)(NC(=O)COc2c(F)cccc2F)C1(C)C Cc1ccc(CC(=O)N(C)CC2CCN(C(c3nscc3C)=O)CC2)c(F)c1 O=C1CC(C(N2CCC(C3CCCN3C(=O)CCCCC3CC3)C2)=O)CCCN1 NC(=O)CCC(=O)N1CCC(NC(=O)C=CCOC2CCOCC2)C1 c1(C(N(C2CCCC(NC(c3ccc(CCC)s3)=O)C2)C)=O)cc(N)nc(Cl)c1 C(=O)(CCCCCC(=O)NC1CCCC1NC(=O)C(C(C)O)N(C)C)OCC C(C1CCOCC1)=CC(=O)N(CC(C(=O)NCC(CC)n1cccn1)C)C CC1CC(NC(c2ccc(C(C)(C)C)cc2)=O)CN1C(=O)Nc1cccc(Cl)c1 S(=O)(=O)(c1c[nH]ccc1=NC1CC(N)CC1(C)C)N(C)CCOCC1CC1 c1(OC)cc(Cl)c(C(N2C(C(N3CC4CCC3CC4)=O)CC3CC23)=O)cc1OC N1(C(c2ccc(C#C)o2)=O)CC(NC(C2CC(=O)N(OC)C2)=O)CC12CCC2 C1(C)(C(=O)OCCC)CC(F)(F)C1.C12CCN(C1)C(=O)C(C)CNC(=O)CC2 Cc1ncnc(C)c1CCNC(=O)NCC1C=CCOC1 C1(O)(COC)CCN(C(c2n[nH]c(C)n2)C(=O)NCC2CCCO2)C1 c1(OC)ccc(OCC(=O)NCC2CCCN2C(=O)C(C)n2ccnc2)cc1 CC1(CNC(C2(C)CC2Br)=O)CCCN(C(C2CC(=O)N2)=O)C1 c1(C(N2C3C(NC(c4cc(C)cc(Cl)c4)=O)C(C3)C2)=O)c[nH]c2nccc-2c1 C1(NC(C(C(CC)O)C)=O)CN(C(c2cc(-c3ccco3)[nH]n2)=O)CC(C)(C)C1 N1(CC)CC(C(=O)NCC(n2cc(CC3CCCC(=O)C3)nn2)C)CCC1=O c1(OC)ccc(=NC(=O)C2CC(F)(F)CN2Cc2ccnc(OC(F)F)c2)[nH]n1 CC(O)CCCCCC(=O)N1CC=C(CNC(C2CC(C(C)C)=NO2)=O)CC1 c1(C(C2CC2F)NC(CNC(=O)Cc2ccsc2)CO)ccc2c(c1)CCCO2 C1(C(=O)NC2C(CC)C2)CCC(NC(c2ccnn2C2CC2)=O)CC1 Cc1sc(C)c2sc(C(=O)NCC3CCCCC3NC(=O)CC(F)(F)F)cc12 c1(C(CNC(C(C)(C)OC(C)C)C2CCCC2)(C)C)cccc(C(F)(F)F)c1 C(C(C)(C)CNC(c1cnn(-c2ccccn2)c1)=O)N(C(=O)CN1CSCC1=O)C N1(C(C(=O)NCC(F)CO)=O)CCc2ccccc2C(O)C1 CC(C)CCC(=O)NC1(C)CN(C(=O)CCN2CCCCC2C)C1 c1(NC(C2C(C(=O)Nc3ccc(Cl)cc3I)C2)=O)[nH]nc2ncccc12 C1(NC(CS(=O)(=O)NC(C)(C)C)=O)CN(C(=O)C=Cc2cc[nH]c2)CCC1O c1(C(=O)NCC(C)NC(=O)CCNC(c2ccc(O)cc2)=O)cn(C)c(C(F)F)n1 N1(C(c2c(SC)scc2)=O)CCOCC(NC(=O)CN2CCCC2C)C1 CCC(CC)CC(F)C(=O)NCc1nocc1C(N1CCCC(C)C1)=O CC(CC(=O)N1CCN(C(=O)Cn2cccn2)C2COCC12)CC(F)(F)F c1(OCC)c(C(N2CC(CO)(NC(c3cc(C)cc(C)c3)=O)C2)=O)cccc1F c1(CNc2ccc(NC(C(CSC)(C)C)=O)cn2)cc2cnccc2[nH]1 c1(OCCCC(=O)NCC2CCCCC2NC(=O)COC(F)F)cccc(F)c1 C1(N(C(CCOCCC)=O)C)CCN(C(c2csc(COC)n2)=O)CC1C C(N=c1nc(N2CCC(O)C(F)C2)c2c(F)cccc2[nH]1)c1nccc(CC)c1 N1(C(C2C(C)CCCC2)=O)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CCC1C N1(C(C=C(C)c2ccccc2)=O)CC2CCC(N(C(=O)CCF)C)C2C1 C1(NC(C(CC)F)=O)CC2(C1)CN(C(C1CCCN(C(C)=O)C1)=O)C2 CC(CNC(c1cccnc1-c1ccccn1)=O)(C(F)(F)F)c1ccccc1 N#Cc1cncc(CC(N2CCCC2CNC(c2ccc(F)cc2Cl)=O)=O)c1 O=C(C1=CS(=O)CCC1)OCCn1cnc(C(=O)NCc2ccccc2)c1 N(C(=NCCCC1CCCCO1)NCC1(C)CCCCC1)C(c1cccs1)C Cc1nc(C2CC2)sc1C(=O)N(CC(C)NC(C1CC12CCCC2)=O)C C1(C(=O)NCC2CCCC2CN(C)C)(NC(CC=CC)=O)CCCCC1 N1(C(CCCOC(C)=O)=O)CC2CC2C1C(=O)NC1C(=O)OCC1CO C#Cc1cncc(C(N2CCC(CCC(=O)NC(CC)(CC)CC)C2)=O)c1 N1(C(CCOCC#C)=O)CCC(NC(=O)CCc2cscn2)C2(CCC2)C1 O(NC(=O)C(C)N(C)C)c1c(CCCC)nsc1 CN1C(=O)Cc2c(NC3CC34CCN(C(c3cnc(O)[nH]3)=O)CC4)ncnc21 CCC(C)C(C(=O)NC(C(=O)Nc1cccc(C(F)(F)F)c1)C1CCCC1)N(C)C N1(C(C(c2ccccc2)NC(C(C)C(F)(F)F)=O)=O)CCC2(CCCCO2)C1 N1(C(C(CC)COC)=O)CCN(C(=O)C2=CCSC2)CC1CCOC N1(C(c2n(CC)ncc2)=O)CC(C(N2CC(n3ccnn3)C2)=O)CC12CCC2 N1(C(C(C2CCC2)OC)=O)CCN(C(C2CC3(CCC3)C2)=O)C(C(C)C)C1 CN1CCN(C(C2CC3CC3N2C(=O)Cc2cccc(F)c2)=O)CCC1=O CC1CCCc2cc(C(N3CCC(CC(C)NC(=O)C4CC4)CC3)=O)nn21 C(=O)(CC(C)CC(=O)OC)NC1(COC)CN(C(=O)C(C)(C)CO)C1 c1(CN=C(NC(=O)C(C2CCOCC2)O)NCC(F)F)cc(O)cc(F)c1.CCC CCC(O)C(C)(C)C(=O)N1CCCC(C)(CNC(=O)CCc2cc(C)nn2C)C1 c1(C(N2C(C(N3CCCC(C#N)C3)=O)CC3CC32)=O)cc2ncccc2[nH]1 Cc1cc(Cl)c(C(=O)NC2CC3CC2N(C(=O)CCc2cn[nH]c2)C3)cc1F Cc1cc(C(=O)NC2CCCCC2CNC(C2CCN2C)=O)ccc1F C1(NC(C2CCOC2)=O)(CO)CCCN(C(=O)CCC2CCCCO2)C1 c1(C(N2CC(C(C)(C)O)(CNC(c3nc(C)c(C)s3)=O)C2)=O)ccc(Cl)nc1N N1(C(C2CCN(C)CC2)=O)C2CCCC1CC(NCc1sc(Cl)nc1Cl)C2 c1(C(=O)NC2C(CCC)CN(C(C3C=CCC3)=O)C2)cnc(C)cc1C C12(CNC(=O)Cc3cnc[nH]3)CCC(C1)N(C(c1cc(F)ccc1F)=O)C2 C1(C(=O)NC(c2c(C)cccn2)C)(NC(c2ccnc(O)n2)=O)CCC(C)(C)C1 CC1CC(C(=O)NCC2CN(C(c3occc3-c3ccccc3)=O)C2)CO1 C1(CNC(c2cnc(C#N)s2)=O)CN(C(C2CC23CCC3)=O)CC12CC2 Cc1cc(NC(=O)CNC(C2(CSc3csc(C)c3)CCC2)=O)no1 CC(C1C(=O)N1)C1CCCCC1.C1(C#N)(OCc2ccccc2)CCC1.C(COC)N c1(C(=O)NC2CCC(NC(C3(COC)CCCO3)=O)CC2)cc(=O)c(O)c[nH]1 c1(OC)cc(NC(C2CCCC2NC(c2cccnc2)=O)=O)c(F)cn1 Cc1oc2ccccc2c1C(=O)NC1CC1NC(=O)CCc1cc[nH]n1 N1(C(CCCCC)=O)CCC(C2CCN(C(=O)C(c3cnn(C)c3)O)CC2)C1 Cc1cc(C(N2CCC(C(C)(O)CNC(=O)C(C)(C)C)CC2)=O)cnc1O C1(NC(C(COCC)C)=O)CCCCN(C(=O)Cc2ccc(OC(C)C)cc2)C1 c1(NC(=O)Nc2nccc(Br)n2)ccc2[nH]cc(CN3CCN(CC)CC3)c2c1 C1(CC(=O)NCc2n(C)cnn2)CC(O)CN1C(=O)CC1CC(C)(C)CO1 C=CC(C)(C)C(=O)NCCC1(NC(c2cnn(CCC)c2C)=O)CC1 C(C(=O)N1CCCC1C(C)(C)NC(=O)Cc1cc(C)no1)(C(C)C)SCC C1(C)(CNC(c2n[nH]c(C)c2C)=O)CN(C(=O)CCCCCF)CCO1 C(=O)(CCS(C)=O)NC(c1cn(CCCC(=O)OC(C)(C)C)nn1)C.C(=O)O c1(C(N2CC3C(CNC(c4ccn(CC#N)n4)=O)(C3)C2)=O)cccc2nc[nH]c12 CCCC(C(=O)NCCCc1cc(C)no1)NC(c1ccc(C#N)o1)=O c1(C(N2CCC(C(C)NC(=O)Cc3cc[nH]c3)C2)=O)c(F)cc(C#N)cc1F C(c1csc(Br)c1)=CC(N1C(CNC(CC2(C)CCC2)=O)CC1)=O c1(OC)ccc(C(F)(F)F)cc1CNc1ccsc1C(N1CC2CC2C1C#N)=O c1(C(C(=O)CCN2CCCC2=O)=O)cn(C2CC2)cn1.C(CCN)NCCO C1(C)(OC)CN(CCNC(=O)NCCNc2ccccc2)C1.OCC N1(c2nnc(CC)o2)CCN(C2CCCN(C(C3CC(=O)N3)=O)C2)C(=O)C1 C(CCC(C)C)(C(=O)NCCC(C)(O)C1CC1)NC(c1ccc(C)[nH]1)=O c12ccccc1S(=O)(=O)Nc1ncc-2cn1.C1(C(=O)OC)CCCN(C(C)=O)C1 CC1CN(C(C2CSC2)=O)CCC1NC(=O)C1=CSCS1 CC1(CCC(=O)NC2CC3C=CC2C3)CCCN1C(=O)CCN1CCCC1=O CC1CN(C(C2(C)CC(=O)C2)=O)CC(C(=O)NC2(CF)CC2)O1 N1(C(c2cnc(OC(C)C)c(Cl)c2)=O)C2CCC1CN(C(=O)CCC(N)=O)CC2 N1(C(C2CC(=O)NC2)=O)CC(NC(=O)COc2cccc(F)c2F)C2(CC2)C1 C1(NC(CCCC(C)O)=O)CCCOC12CCN(C(=O)COc1ccon1)CC2 CC1(C)CCC(C(N2CC(F)(C#N)C2)=O)CN1C(C1C2CC3C(C2=O)C13)=O C1(C)(CNC(C(C2CCC(=O)NC2)C)=O)CN(c2nc(Cl)c(C#N)s2)CCO1 c1(CNC(c2n(CC=C)nnn2)c2ccco2)ccc(OCC)cc1 C1(CNC(c2cc[nH]c2)=O)COCCN1C(C1(c2ccc(Cl)nc2)CC1)=O C(=O)(C(CC)C(=O)N1CCC(C)(C(=O)N(CC(O)CO)C)CC1)OCC C1(C2CC2)(CNC(CC)=O)CCN(C(c2cnn(C)c2N)=O)C1 C1(NC(c2cn(CCOC)nc2)=O)CC2(CCN(c3ccnc(C4CC4)n3)C2)C1 N1(C(CSCC#C)=O)CCN(C(C2CCC(NC(C)=O)CC2)=O)C2COCC12 N1(C(c2nccc(CNC(=O)C(O)CC(F)(F)F)c2)=O)CC2CCCC2C12CC2 c1(C2C(C(N(C3CCN(C(c4sncc4Br)=O)C3)CC)=O)C2)ccccc1 C=CCC(C)(C)CC(=O)N1CCOC(C(N2CCC(F)(F)C(O)C2)=O)CC1 N1(C(CC(CC=C)NC(=O)CCCN(C)C)=O)CCC(O)CC12CC2 N1(C(C#CCNC(Cc2c(C)nccc2)=O)=O)CC(C)(C2CCC2)C1 C1(C(=O)NC2CCN(C)CC2)C2CCCCCCC12 N1(C(C(CC)N(C)C)=O)CCCCC1CNC(=O)CC1CC(C)OC1C C1(CNC(C2C(C)C2)=O)CCC(NC(c2ccoc2Br)=O)C1.C1CC(=O)N1 C1(CNC(c2c(CC)ncs2)=O)CC(F)(F)CN1C(C1CCCC(C2CC2)O1)=O C(C(C)(C)C(=O)NC1CC1NC(=O)CCNC(c1ccccc1)=O)OC O=C(CCCCC(F)(F)F)NC1CC(F)(CNC(=O)CC2CC3CCC2O3)C1 C1(CNC(COCCOC)=O)CC12CCN(C(c1cncc(Br)c1)=O)CC2 CC(C)CC(CNC(=O)C(C)CN(C)C)NC(c1ccc(=N)[nH]c1)=O Cc1cc(C(=O)NCC2CN(C(=O)Cc3csc(Cl)c3)CCO2)c(O)c(C)n1 c1(C(=O)NC2C(CC)CN(C(=O)CC(F)(F)F)CC2)ccc2ncc(=O)[nH]c2c1 CC(O)C(F)(F)C(=O)N1CCOC(CN(C)C(c2cncs2)=O)C1 c1(C(N2CCN(C(C#CC(C)(C)O)=O)C(CCN(C)C)C2)=O)ccn2cccc2c1 N1(C(c2n[nH]c(O)n2)=O)CCCC(CNC(=O)C(c2ccc(F)cc2)(F)F)C1 c1(C(=O)NCC2(CO)CCCNC2)cnn2c1NCCC2C(F)(F)F N1(C(C2OCCN(C(C(CC)N(C)C)=O)CC2)=O)CCN(CC)C(C)(C)C1 N(C(=NCCCC(F)F)NCCOCc1cc(C)c(F)cc1F)C(CC)C Cc1nc(Br)sc1C(N1CCC(C)(CO)C1)C(=O)NCCC1(C)CC1 C(=O)(C1=CCCC1)N1CCC(OCC(=O)N(C(C(C)C)C)C)C1 C1(NC(CCSCCCC)=O)CC(CNC(=O)CCCc2cncs2)C12CCC2 c1(C(N2C(CNC(C3(OC)CC3)=O)CC2)=O)cccn(CC(=O)N(C)C)c1=O C#Cc1cc(F)c(C(N2CCC3(C2)CN(C(=O)C(C)(CC)CC)C3)=O)cc1F Cc1onc(CC(N2CCCC2CNC(=O)CCC2CC2(C)C)=O)c1C#N c1(C(=O)NCC(CN(C)C(C2CCOC2(C)C)=O)O)ccc2nc[nH]c2c1 C(=O)(C1CCCc2nncn21)NCC(C(C)C)NC(C(C)NC(CC)=O)=O CN1CCn2nc(C(=O)NCC3(C)CC(F)(F)CN3C(c3cc[nH]n3)=O)cc2C1 c1(C(=O)NC(CNC(c2cc(C)c(C)nc2)=O)(C)C)cc(F)cc2c1NCCC2 N1(C(Cc2cnc(C)s2)=O)CCN(C(=O)C(C)C(C)O)CC1C(C)C N1(C(CC)=O)CCN(CCOC)CC1.C(=O)(C(CC1CCCO1)OC)N(C1CC1)C N1(C(C(C)(C)CCNC(c2ccoc2Cl)=O)=O)C2CCC1CC(F)C2 c1(OC)ccc(CCNC(=O)C(N2CC(c3ccccc3)CCC2C)=O)c(Cl)c1 N1(C(C(C)CS(C)(=O)=O)=O)CC2(CCCN(C(=O)CCOC3CCCOC3)C2)C1 C=CCCC(C)(C)C(=O)N1CCC=C(C(=O)NCc2cn(C)nn2)C1 C1(CCC(=O)NC2CCCC2(F)F)CCN(C(C2CCC(F)(F)C2)=O)CC1 N1(C(CCN(C(C(C)(C)C)=O)CCO)=O)CCCc2cccc(Br)c2C1 N1(C(C2CNC(=O)O2)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)CCO2 Brc1cc2ncnc(N3CCC3)c2s1.c12ccc(cc1)C1(CC1)Nc1scnc1-2 c1(C(N(C)CC2(O)CN(C(C3(C)C(C(=O)OC)C3)=O)C2)=O)c(F)ccc(O)c1F N1(CCNC(c2c(C)onc2)=O)CCN(C(c2cnn(CC3CC3)c2)=O)CC1 N12CCC(CC1)C2=O.C1(C(N(CCCOCCNC(C)=O)C)=O)OCCC1CC c1(C(N2CC(CC(N3CCOC4CC34)=O)C2)=O)cc(Br)cc2[nH]ccc12 CN1CC=C(CC(=O)N2CC3(CCCC3)C2C(N2CCC(CC(N)=O)C2)=O)CC1 c1(OC)cccc(Br)c1C(N1CC(O)(CNC(c2cc(C)nc(C)c2)=O)C1)=O CC(C)(C(=O)NC1CCCN(C(c2c[nH]ccc2=O)=O)CC1)C(F)(F)F c1(OC)cc(N2CCC(N3CCN(CC4CCC(F)(F)C4)CC3)CC2)ncn1 C1(C(=O)NCC(O)C2CC2)CC=CCC1NC(c1[nH]nnc1C1CC1)=O C(CC)(CC)(CCNC(=O)CN(C)Cc1ccccc1C)NC(CCCC)=O C1(O)(C(CC)C(=O)NC2CCC2CNC(C2(C(=O)NC)CC2)=O)CCCCC1 c1(C(=O)NC(C(C)C)CCNC(c2cccnc2CO)=O)cccc2c[nH]nc12 CC(=NO)C1CC(C(=O)NCC2CCCCN2C(=O)C(C)C2CCCO2)C1(C)C c1(CNC(C)C(N2CCOCC2)=O)nccc2c1CNCC2 C1(CC=C)(C(=O)N(C)Cc2ccc(C)nc2)CCN(C(=O)C(C)OCCOC)C1 C1(C(N2CC(O)(CNC(C3(NC(C)=O)CCCC3)=O)C2)=O)CCOC2(CCC2)C1 C(=O)(C(C)(C)C(F)F)N1CCC(C(CNC(C(C=C)OC)=O)O)CC1 C(=O)(CC(C)(C)C(F)F)N1C(CNC(c2cc(C(C)C)[nH]n2)=O)CC(C(C)C)C1 C1(C(N2CCC(N(CC(C)C)CCO)C2)=O)CN(C(=O)OC(C)(C)C)CCCO1 C(=O)(CC(F)(F)C(F)(F)F)NCCCC(c1cccs1)NC(=O)CC(=O)NC1CC1 c1(C(N2C3CC(N(C(CCC#CC)=O)C)CC2CC3)=O)ccc(F)c2occc12 N1(c2nccc(N3CCC(NC)CC3)n2)CC(C)CC(C)(C)C1.CC1CNC(C)(C)C1 C#Cc1ccc(Cl)c(NC(N2CCS(=O)C(C)C2)=O)c1 Cn1nc(Br)c2ccc(C(=O)NC3CC3C(=O)Nc3ccc4nc(O)[nH]c4c3)cc12 C1(O)(CNC(C2CC(C3CCC3)C2)=O)CCN(C(=O)C(F)CC2CCOC2)CC1 c1(C(N2C(C(N(C)Cc3c(C)occ3)=O)CCCC2)=O)ccc2cc[nH]c2n1 c1(C(=O)NC2(CN(C)C(c3c(Br)ccc(F)c3F)=O)CC2)ccc2c(c1)OCCO2 c1(OCC)ccc(C)cc1NC(N1CCC(C)(NCc2cccnc2OC)C1)=O N1(C(=O)CC=C(Cl)Cl)CCN(C(=O)C(O)CF)C(C2CC2)C1 c1(NS(CC#N)(=O)=O)ccnc(O)c1 N1(C(CSCCCC)=O)CC2C(CNC(=O)CCn3ccnc3C(C)C)C2C1 c1(NC(C2N(C(C(C)NS(CC)(=O)=O)=O)CCC2)C)cc(Cl)ncn1 CC(O)C(C)(C)C(=O)N1CCC(C(=O)NCc2n[nH]cc2C2CC2)C1 CCCCC(CC)CC(=O)NCCC(O)CNC(c1cc(-c2ccco2)no1)=O Cc1ccc(NCC(=O)NC(C)CCNC(C2CC(C(C)C)C2)=O)cc1 Cc1cc(C)c(CC(=O)NCC(C)N(C)C(c2cnc3nccn3c2)=O)c(O)n1 C(C)(CCCCNC(=O)CCC(C)c1ccccc1)NC(CN1CC(CC)C1)=O N1(C(CNC(N)=O)=O)CC2CCOC2(CNC(=O)C(F)(F)c2cccnc2)C1 N1(C(COCc2cccc(C)c2)=O)CC2CCC1C(NC(c1ccnnc1)=O)C2 c1(OC)cccc(C(=O)NC(C)C(C)(C)NC(=O)C(C2CC(F)(F)C2)O)n1 c1(C(N2CC(O)(C(C)(C)CNC(c3cnco3)=O)C2)=O)ccccc1CO N1(C(C(C)=CC)=O)CC(NC(=O)C(O)Cc2ccccc2)C(n2cccn2)C1 c1(C(=O)NC2CCC(NC(CC(C)(C)SC)=O)C2)cccn2c(O)nnc12 Cc1cc(C(=O)OCC(=O)O)nn1C1CCC1.C(C)(C(=O)OC(C)C)NC(N)=O CC1(C)CN(C(c2cc(Cl)c(F)c(Cl)c2)=O)CC(C)(C)C1NC(=O)C1=CCCS1 Cc1cc(C(=O)N(CCCN(c2ncc(Br)c(O)n2)C)C)cc(O)n1 C=CCC(CNC(c1cscc1C(N)=O)=O)NC(C1CC1C)=O Cc1nc(O)[nH]c1C(=O)N(C(CNC(c1cc(O)nn1C)=O)C1CC1)C c1(C(=O)NCC2C(NC(CCn3ccc(C)n3)=O)C2)ccc2c(c1)C(=O)CCC2 C1(C(=O)NCC(CN(CC)CC)F)CCCN1C(=O)NC1CC1 C1(NC(C(C)Cn2ccnc2)=O)CCN(c2ccnc(Cl)n2)CC1C c1(CC)cc(C(=O)NC(Cn2cccn2)C(=O)NCC(C)(C)CC2CC2)no1 CCCCC(C(=O)NC)NC(=O)C(C(C)C)NC=O.C1CCOCCN1 C(C(C)(O)CNC(=O)C(CO)N(C(C)=O)CNC(=O)C(C)Cn1ccnc1)OC C1(C(=O)NC2CN(C(CCCCOC)=O)C2)CC(C)(C)CCO1 C#Cc1ccc(C(N2CCCC(CNC(=O)C(C)OC(C)=O)C2)=O)cc1C CS(=O)(=O)C1CCCC(NCc2nc3ccc(Br)cc3o2)C1 N1(C(C2(C=C)CC2)=O)CCCC(C2CCN(C(=O)C3=CCC3)C2)C1 C1(CC(=O)NC(C)CCCNC(=O)C=CC2CCCN2C)CN2CCC1CC2 N1(CC(=O)NCCC(C)NC(=O)C(C(C)(C)C)N(C)C)CC(=O)N(C)C1=O N1CC2CCCC2(NC(C2C3(C2)C(=O)NC3)=O)C1.c1(COC)ccccn1.C1(C)CC1 C(C1=NOC2CN(C(C3CCOCC3)=O)CC12)NC(c1cc(C(F)(F)F)c[nH]1)=O CON=CC(=O)NC(CNC(C1CC1(C)C)=O)C1CCC1 Cn1ncc(C(=O)OC2CCC(OC3CCC(=O)N3)CC2)c1-n1cccc1 c1(C(=O)NC2(CNC(=O)C(F)(F)c3ncc[nH]3)CCOC2)cccc(OC(F)F)c1 C(CCN=C(NC(C)C)N1CCC(F)(c2ccccc2Cl)C1)=CC Cc1ccoc1S(=O)(=O)NC(C1CNCCOC1)=O C(=O)(C(C)(O)CNC(=O)C(c1cnn(C)c1)NC(c1nnsc1C)=O)OC C(=O)(C(CC(F)(F)F)c1ccccc1)N1CC2C(COC(C)(C)C)C2C1 c1(C(=O)NCC(CC)(C)NC(c2nc(Cl)sc2C)=O)c(C)cc(C)cc1C C1(CCCC)CCCN1C(=O)CNC(C1(OC(C)=O)CC1(C)C)=O c1(OC)cc(C(=O)NC2CCCCN(C(c3ccsc3)=O)C2)c([N+](=O)[O-])cc1F CON=C(C(=O)N1CCOCC(NC(=O)CCc2ccccn2)C1)c1ccco1 C1(NC(c2ccc(CCC)[nH]2)=O)CCC(NC(c2nscc2C)=O)CC1 N1(C(c2cc(C)sc2C)=O)CC=C(C(C)(C)C(=O)N2CC(C3=NOCC3)C2)C1 c1(N(C2CN(C(C(C)n3cnnn3)=O)C2)C)ncncc1Cl c1(C(=O)NCCC(=O)NC2CC3CCCC3C2)ccc2ccccc2c1 C12(C(N3C(C4(NC(CCC#C)=O)CC4)CCC3)=O)CCC(N(C)C)(CC1)CC2 C1(CC(=O)NC2CC(CCNC(C(CC)F)=O)C2)Cn2ccnc2NC1=O c1(CC(N2C(CCCNC(C3CC=CCO3)=O)CCC2)=O)ccc(O)c(F)c1 c1(C(=O)NCC2CC(F)(CNC(C(CC)C(=O)OC)=O)C2)cc2scc(C)c2[nH]1 C1(NC(c2c(C)scn2)=O)CC(C)CN(C(c2cn(C)nc2Br)=O)C1 c1(C(=O)NC2CC(CC(=O)N(C)CC3(O)CCC3)C2(C)C)c[nH]c2ccccc12 c1(NCC(C)N(C(=O)CCc2cc[nH]n2)C)nc(Cl)nc2sccc12 C(=O)(CC1=CCOCC1)NC1CCC(CCC(NOCCCOC)=O)C1 C1(NC(c2c(C)[nH]nc2C(F)F)=O)CC(C)CN(C(=O)C(O)CN2CCOC2)C1 c1(CC(=O)NC2CC(C)(NC(CCC(=C)C)=O)C2)ccc(Cl)cc1C N1(C(c2cc(C)[nH]n2)=O)CCC(C(=O)NC(C2CCCC2)C)(C(C)C)C1 c1(OC)cc(F)ccc1C(N1CC2CC2(CNC(=O)CSc2nc[nH]n2)C1)=O C1(CNC(CS(=O)(=O)N(C)C)=O)CCC2(CN(C(c3cccc(F)c3N)=O)C2)O1 C1(NC(CSCC(=O)OC)=O)CN(C(=O)CCCN(C)N=O)C2(CCCC2)C1 C1(CNC(C#CC(C)C)=O)(NC(=O)CN(C)S(N)(=O)=O)CC2CCC1CC2 C1(CC=C)(NC(=O)CCCCCCN)CCCN(Cc2noc(C3CC3)n2)C1 C1(C(N(C2CCCCC2)CCOC)=O)CCC(NC(c2cnc(Cl)s2)=O)CC1 c1(NC(c2ccco2)=O)ccc(NC(c2ccccc2CC(F)(F)F)=O)cc1Br C1(NC(c2ccc(COC)o2)=O)CC2(CCCN(C(=O)COC3CCOC3)C2)C1 N1(C(C(C(CC)CC)C)=O)CC2(NC(c3cncc(N)n3)=O)CCCC2(F)C1 CC(CC(=O)NC12CC(C(=O)NCc3nncn3C)(C1)C2)CC(C)(C)C C(=O)(C(F)CC(C)(C)C)NCC1CC(CNC(c2c(CCC)cccc2)=O)C1 c1(C(=O)NCC(F)(F)CC2CC2)ccc(F)c(Br)c1F C1(Cc2ccccc2)Cc2cccc(F)c2O1.c12csc(n1)CSN(CC)C2 c1(CC)nc(Cl)cc(=NCC2(C)CCN(C(c3cc(C)nc4ncnn34)=O)C2)[nH]1 c1(OC)nc(NC(=O)NCC2CCCCC2C(F)(F)F)sc1C c1(C(N2CCC(C)(CNC(=O)C3=NOCC3)C2)=O)c[nH]c2cc([N+](=O)[O-])ccc12 c1(C(=O)NCCCC2(NC(C3ON=C(C)C3)=O)CC2)cccc(C)c1F C1(CNC(C(CC)C)=O)CC2CCC(C1)N2C(C1CCS1(=O)=O)=O C1(C)(C(=O)N)CC=CC1.C1(C(NOCC=CC)=O)CC(CCCCSC)C1 c1(C(N(C)CC)=O)ccc(C(=O)NC(C)C(C)NC(C2(N=[N+]=[N-])CC2)=O)cc1 CN1CC(C(=O)NCC23CC(NC(c4csc(Cl)n4)=O)(C2)C3)CC1=O C(C(C)CC(C)C)C(C1(COC)CC1)SC1CCCCC1C1CCCO1 Cc1noc2cc(C(N3CC(NC(c4cccc(N)c4)=O)C3)=O)ccc12 C(=O)(C(O)CC(F)F)N1CCC(N2CCN(C(C3CC(C(=O)OC)C3)=O)CC2)CC1 C12CN(CC1NC(C1CCN(C(=O)CC)C1)=O)C(=O)N2.CCC(=O)OC(C)C C=CC(C)(CC)C(=O)NC1CCC(NC(=O)Cc2cnccc2C)C1 N1(C(C(C=C)O)=O)CC2(C1)CN(C(=O)C(O)Cc1cnc[nH]1)CC(C)(C)O2 Nc1cc(C(=O)NCC2CCN(C(c3cnc4sccn34)=O)CC2O)ccc1F CC(C)(C)C(CC(=O)N1CCC(NC(=O)COC(F)F)C2(CCC2)C1)C(F)F CCC(C)(C)C(C)CC(=O)NC1CCCC(NC(=O)CCCOC)C1 c1(CNC(C(CCC)C)(C)c2nnnn2C)cn2cc(C)ccc2n1 c1(C(CCC)N(C(=O)C(C)NC(=O)C(C)C)C)ccc(Cl)cc1 CCC(O)C(C)C(=O)NCC(C1CCCC1)NC(c1n[nH]cc1Br)=O N1(C(c2c(C(C)C)occ2)=O)CCC(F)C(NC(=O)C=C2CCCCC2)C1 CC(CC(F)F)C(=O)NCC1CC(F)CN1C(c1coc(CO)c1)=O c1(C(N2CCC(NC(CCOCCC)=O)C2(C)C)=O)cc(Cl)cc2c1CCC2 CN1CC2(CC(NC(c3occc3CNC(C3CN(C4COC4)C3)=O)=O)C2)C1 N1(C(CCNC(=O)OCC)=O)CCCC(N(C(=O)C(C)(COC)OC)C)C1 C1(NC(CCC=CCC=C)=O)(CF)CCN(C(c2snnc2C2CC2)=O)C1 C1(CNC(C(CC)N(C)C)=O)CC2CCC1N(C(c1ccc(C#N)c(Cl)c1)=O)C2 N1(C(COCCOC)=O)CCC(CCNC(c2ccc(OC)cc2Cl)=O)CC1C CCC(CC(=O)NCCC1CC(NC(=O)C(C)NC=O)C1)SC C(C(C)(C)CC(=O)N1CCN(C(C2CC2F)=O)CC1CO)OC1CCN(C)CC1 C1(CNC(c2c(Br)nc(C)s2)=O)CN(C(=O)CN(C)C)C2(CCC2)C1 c1(CN2CCCN(C(c3c(C)n(C)nc3)=O)CC2)csc2ccccc12 Cc1[nH]c(C(=O)NCCOC(C)(C)C)c(C)c1C(=O)Nc1ccc(Br)nc1F c1(C(C2CCN(C(c3cn(-c4cn(C)nc4)nn3)=O)C2)=O)cnn2ccncc12 C12(CC(=O)NCCCCNC(=O)CNc3ccccn3)CCCN1CCC2 N1(C(CCN(CC)CC)=O)CC(N(C)C(c2ccc(C)cn2)=O)C(O)C1 c1(C(=O)NCC2C(CNC(C3CCN(C)CC3)=O)C2)c(O)ccc(Cl)c1F c1(NC(=O)CC2CC2)ccc(-n2cnnn2)cn1.Cc1nnnn1C c1(NCC#CC)ncc(S(=O)(=O)NC(C)CCOC)cc1Cl c1(OCC(=O)NCC2N(C(c3n(C(C)C)ncc3)=O)CCC2)cc(F)cc(F)c1 N1(C(C2C(CC)CCO2)=O)CCC(C2(O)CN(C(C3CC(=O)N(C)C3)=O)C2)CC1 N1(C(c2c(C)coc2)=O)CCC(C(=O)NC2CCCSCC2)CC1 C1(C(C)C)CCN1C(C(=O)NC1COC1)c1cccs1 C1(C2CCCN(c3nccc(Oc4ccccc4)n3)C2)(NC(C=C(C)Cl)=O)CC1 CC1(C)CN(C(c2ccnc3ncsc23)=O)CCC1NC(c1cccc(Cl)c1)=O c1(C(=O)NC2CCCC(CNC(C3CCCCC3)=O)C2)cc2occc2[nH]1 C#CCCC(C(=O)NCCOCCCN(C)C(C1C2CC(=O)CC12)=O)N(C)C C=CC1(CC(=O)NCCCc2ccccc2)CN(C(C)=O)C1 c1(C(=O)NC2C(N(C)C)CN(C(=O)C(=O)N(C)C)C2)nc(Cl)ccc1N c1(NCC(O)CN2CCOCC2)cccc(C2(O)CCC2)c1 c1(C(=O)NCC2CCCC(CNC(=O)CCCCCF)C2)cc2n(c1)CCCC2 CN1CC(C)(C)CC1CC(N1CCCC(O)(CNC(C2(C)COC(=O)N2)=O)C1)=O C1(NC(CC2C(CNC(C(c3ccn(C)c3)C)=O)C2)=O)CC(C)(C)C12CCC2 c1(C(=O)NCC(CN(C(=O)CCC2CCC(=O)N2)CC)(C)C)cc(O)nc(Cl)c1 C1(C(=O)NCCN(C(C(C)(C2CC2)OC)=O)C)CCC(CCC(C)C)CC1 C(CC(=O)Nn1ccccc1=O)C1CCCN(C(CSCC#C)=O)C1 C1(CNC(CSCCCC)=O)C(C)CCN1C(=O)CCC(=O)N(CCC)CC C1(C(C(=O)NCCCOC)N2CCC2C(=O)OC)CCC(C(C)(C)C)CC1 CC1C(NC(=O)CC2CCCCCCC2)CCCN1Cc1ccsc1 CC1Cc2cc(Br)ccc2CN1C(c1ccc(=O)n(-c2ccccc2)n1)=O N(C(=NCc1ccnn1C)NCC1(C)CCCOC1)CC1(NS(C)(=O)=O)CCC1 C1(NC(c2n(CC)ncn2)=O)CCCCC1Cn1cc(CCN2CCCC2)nn1 N1(C(c2c(Cl)ncc(OC)c2)=O)CCN(C(=O)CC2CC3(CC3)CO2)CC(O)C1 c1(C(N(CC(C)C#N)C)=O)ccnc(CNC(=O)OC(C)(C)C)c1 C1(CCNC(c2c(C)nc(COCC(C)C)s2)=O)CCN(C(=O)CO)CC1(F)F C1(N(C(=O)C(F)C2CCC2)C2(CC(N3CCCCC3)=O)CC2)COCC1CO C1(CNC(C(C=C)OC)=O)CN(C(=O)Cc2cnn(C)c2)CC1(F)CO CCCC(C(=O)NCC1CCCCN1C(c1cc[nH]n1)=O)OCC C1(CNC(CCCCC=C)=O)CCC(C)(C)CN1C(=O)C(C)C(C)COC c1(C(N2CC3CCC3(F)C2)=O)cc(I)cc(I)c1 c1(N2CCC(NC(c3ccn(CC)n3)=O)C23CCC3)nc2ccc(OC)nc2s1 CC(CO)(CO)C(=O)NCc1ccc(-c2ccccc2)o1.C12(O)CCCN(C1)C2 C=Cn1ncc(C(=O)NCC=CC(=O)N(C)CC2(C)CCC2)c1N C(=O)(CCCCC(=O)NCC1(O)CC(CNC(C2CCC3(CCC3)CC2)=O)C1)NC c1(C(=O)NC2CCN(C(c3ccncc3)=O)CC2O)ccn2nncc2c1 N1(C(CCCOC(CCC)=O)=O)CC(NC(c2nccnc2N)=O)CC(C)C1 N1(CC(=O)N(CCC(C(C)C)NC(C2(C)CC=CCO2)=O)C)CCP(C)(=O)CC1 C1(C)(NC(C2CC(CNC(C3C(C)=CCS3)=O)C2)=O)CCCCCC1 C1(N(C(=O)C(C)(C)c2cccs2)C)CCCCC1N(C(=O)Cn1nnc(=N)[nH]1)C c1(C(=O)NC2C(NC(c3n[nH]c(C)c3C)=O)CC2)ccc2nsnc2c1 c1(C(=O)NCCCN(C(=O)Cc2cncnc2)C)nccc2ccn(C)c12 C1(N(C(=O)CSS(C)(=O)=O)C)CCCN(CC2C(c3ccccc3)C2(F)F)CC1 c1(NCc2cn(CC)nn2)ncc(C)cc1S(=O)(=O)NC1C(C)C1(C)C c1(CCOCC)nc(C(=O)N(CC(C)(C)NC(C2CCC(N(C)C)C2)=O)C)co1 C1(CC(=O)Nc2c(C)nsc2)CCCN(C(=O)CC(C)C)C1 c1(C(=O)NCCC2(NC(C3=C(C)OCC3)=O)CC2)ccc2c(c1)C(=O)N(C)C2 c1(C(N(CC)Cc2cc(C)on2)=O)cn2c(n1)CCN(CC1(CC)COC1)CC2 C(=O)(CS(=O)CCC(F)(F)F)NCCC1CN(C(C2C(OC)(OC)CC2)=O)C1 N1(C(c2c(CC)ocn2)=O)CCCC2CN(c3cnc(C#N)c(C#N)n3)CCC12 C1(NC(C2C(CC)CCC2)=O)CCCC12CCN(C(=O)C(C1CC1)SC)CC2 CCC(C)(CNC(=O)C(C(C)C)OC)C(=O)NOCC=CCl c1(C(=O)NCC2C(NC(c3coc(Cl)c3)=O)C2)cc2ccc(Cl)cc2s1 c1(C(=O)NC(CCCNC(CC=C=C)=O)C)c(OC)cccc1C(F)F Cc1occc1C(=O)NCCCOCCN(C)C(C1CC(C)(F)C1)=O C1(NC(C2(N(C)C)CC2)=O)CN(C(=O)CCn2ccnc2)CC2(CCC2)C1 c1(C(N2CC(C(C)NC(c3cc(SC)c(C)o3)=O)OCC2)=O)cncc(Cl)c1Cl N1(C(c2c(OC)c[nH]n2)=O)CC2COCCC2(NC(c2cc(N)ccc2Cl)=O)C1 C1(CC(=O)NCC(CCOC)NC(C2(C(C)C)CCCO2)=O)CCN(OC)CC1 Cc1ccc2nonc2c1C(=O)NC1(CO)CCN(C(C2CCOC2)=O)C1 C1(CC)CN(C(=O)C(F)(F)c2cnn(C)c2)CCC1CNc1cc(O)nc(C)n1 c1(C(=O)NCCC2CC(NC(C3CC3(F)F)=O)C2)ccc(=O)n(-c2nccs2)n1 N1(C(c2nc(OCC)sn2)=O)CCC(NC(=O)CCSCC(C)C)C(CO)CC1 Cc1cccc(-n2cc(CNC(=O)CC3CCC4CC34)cn2)c1 N1(C(C)=O)CCC(CC2(OC(=O)Nc3nc(C(C)(C)C)cs3)CCC2CC=O)C1 CC1CCCCN1CCC(=O)NC1CCC1CNC(c1ccsc1Cl)=O c1(C(=O)OC)ccc(Br)cc1S(=O)(=O)N1CC(c2cccc(F)c2)C1 c1(CC(=O)NCC(CNC(C(C(CC)O)C)=O)O)noc2ccccc12 CCCC(CCCNC(c1nc(Br)sc1C)=O)NC(C12CCC(C1)C2)=O C(CC(C(=O)NCC(=C1CCCCC1)F)NC(C1COCCN1C)=O)SC N1(C(c2nn(C)c(F)c2)=O)CC(C2CN(C(C3CC3c3ccnn3C)=O)C2)C1 c1(NC(C2(CC)N(C(C(CC)N(C)C)=O)CCC2)=O)ccc(OC)cc1F c1(OC)c(NC(=O)NCC2CC2c2cccc(C)c2)c(C)nn1C N1(C(C(CCC)F)=O)CCC(C(=O)N(C)CCC2CC2)C12CC2 C1(CNC(C(C)(F)F)=O)CCN(C(C2CC2C2CC2C)=O)C1(C)C c12ccc(nc1)[nH]2.C1(C(CNC(=O)COC(C)=O)OC)CCOCC1 c1(OC)ccc(F)cc1C(c1nnnn1C)NC(CC(C)C)CCc1ccccc1 c1(OC)cccnc1C(N1CCOCC1Cc1cn(CCCN(C)C)nn1)=O C(C(C(=O)N(C(CO)C(C)C)C)C(C)C)NC(C(COC)COC)=O Cc1cccn2ncc(C(N3CCCC3C(=O)N(CCC(N)=O)C)=O)c12 N1(C(C(=O)NC(c2ccc(Cl)s2)COCC)=O)CCC(CC(C)C)CC1 c1(C(N(C2CN(C(CC(COC)C)=O)CC23CC3)C)=O)ccc([N+](=O)[O-])n1C N1(C(c2ccnc(Cl)c2F)C(=O)NCc2cccnc2)CCOCC(C2CC2)C1 C(=O)(C#CC1CCOCC1)N(CCCCC(=O)NCC1(O)CCCOC1)C c1(C(=O)NC(C2CCN(C(CNC(=O)OC)=O)C2)C)cc2cccc(O)c2n1C C1(NC(Cc2ccc(CC)cc2)=O)CN(C(c2cnnn2C)=O)CC1(C)C c1(C(=O)NCCC2N(C(CC3C(C)(C)C(O)C3)=O)CCC2)ccc2c(c1)COC2 CC(C)CCC(F)C(=O)N1C2CCC1CC(C(=O)NCCN(C(C)C)C1CC1)C2 c1(C(=O)NCCCC(C)NC(C=C(C)c2ccsc2)=O)cccc2nsnc12 N1(C(CC#N)=O)CCN(C(c2csc(-c3ccco3)n2)=O)CC(O)C1 c1(NCc2cccc(C=C)c2)cc2c(F)cc(F)cc2o1 C1(NC(C2C(C)OCC2)=O)CCN(C(C2CC23CC(O)C3)=O)C12CCCCC2 n1(CC(=O)NCC2(CNC(c3c(CC)noc3)=O)CC2)cnc2ccc(C)cc12 N1(CCN(CC=CCNC(C2C(C)(COC)C2)=O)C)CCCNS1(=O)=O c1(C(=O)NC23CC(CNC(c4cc(OC)ncn4)=O)(OC2)C3)cc2[nH]ccc2s1 C#Cc1cccc(C(N2CCN(Cc3ncc(Br)s3)CC2CCOCC)=O)c1 C1(C(N2C(CCCC)CCC2)=O)CN(C(C2(CCOC)CCC2)=O)CC(C)(C)C1 C=CCCCCC(=O)NCCc1n[nH]cc1C(=O)NCC1(O)CCSC1 c1(N(C)C)nc(C(=O)NCC2CC2NC(c2ccsc2)=O)[nH]c(=N)n1 C(CCN=C(NCc1cncn1C)NCC(C)COC(C)(C)C)N(C)CC.CO C1(OC)CN(C(C23CCCC2C3)=O)CC1NC(C1CCC(OC)CC1)=O C1(COCC)CCCN(C(=O)NC2CCC3(c4ccccc4C)CC23)C1.C Cc1ccnnc1C(=O)NCCC(O)C(=O)Nc1ccsc1C(C)C C1(NC(=O)C(c2ccccc2)N2CCC2)CCN(Cc2cccc[n+]2[O-])CC1F N1(C(Cc2c(C)noc2C)=O)CCOCC(C(=O)NC(C)CCO)C1 C1C(CCCC)C(C)(C)CC(=O)N1C(CC)C N1(C(C(C)CF)=O)CCC(C2CCCN(C(C3CCC4CC4CC3)=O)C2)CC1 c1(NC(c2csc(NC(c3ccc(Br)nc3)=O)n2)=O)cccc2ncsc12 c1(C(=O)NCCN(C)C2CC2)ccc(=O)n(C)n1.C1(OC)CN(C)C(=O)C1 c1(CC)ccccc1C(N1CCC1CNC(=O)C(C)(F)c1ccccc1)=O CC(C)C(O)C(C)C(=O)N1C2CCC1CC(NC(=O)C(C)Cc1cnc[nH]1)C2 C(=O)(C(CNC(=O)CC(C)C)CC1CN(C(C2CC2(F)Cl)=O)C1)OC C(=O)(CCCN=[N+]=[N-])N1CC2C(CC(=O)NC(COCCOC)C)C2C1 c1(C(N2C3(CCN(C(C=CCOC)=O)C3)CCC2)=O)ccnc2cc(F)cnc12 N1(C(c2ccc(C)c(NS(C)(=O)=O)c2)=O)CC2CCOC2(CNC(=O)CO)C1 C1(C(N2CCC3(CCCN3C(=O)CC(O)C3CC3)C2)=O)COc2ccccc2O1 CC(CN(C)C)CC(=O)NC1(CF)CCN(C(=O)Cn2cc(C(C)O)nn2)C1 C1(C(=O)NC(CC)(C2CC2)C2CC2)CC1C1CN(C(C2(C#N)CCOCC2)=O)C1 C(=O)(CC1=Cc2ccccc2C1)N(C1CN(C(C2CCCCC(F)(F)C2)=O)C1)C C1(OC)CCC(NC(C2(NC(c3nccn3C)=O)CCSC2)=O)CC1 C1(CNC(CSC)=O)CCCN(C(C2(OC(C)=O)CC2)=O)CC1c1ccccc1 c1(C(=O)OC)ccc2c(c1)CN(C(C1(C#N)CCC1)=O)CC2 C1(C2CN(C(C3C(C)CCN3c3ncccn3)=O)C2)(NC(c2cc(C)[nH]n2)=O)CC1 c1(C(=O)NC2CN(C(COc3cc(C)on3)=O)C2)c(C(F)F)nn(C)c1C c1(C(COC(=O)CCCC(=O)c2ccc(F)cc2)=O)cccc2c1CCC2 c1(C(=O)NC(C)CCNC(C2(O)CC2)=O)cnc2c(=O)[nH]ccc2c1 C(=O)(C1CSc2ccccc21)NCCC1(O)CCN(C(C#CC(C)(C)C)=O)CC1 n1(CC)nc(C(N2CC3C(C(=O)NC4(C)CCC4)C3C2)=O)cc1C(=O)OC N1(C(C2CCC(CNC(c3cncc(F)c3)=O)O2)=O)CC2(CC(CO)CO2)C1 C=CCCCC(C(=O)NCCC(F)(F)CO)NC(c1csc(Cl)n1)=O C1(NS(=O)(=O)NCC(C2CCCO2)O)CCC2(CCC2)OC1 N1(C(C(C)SCCCC)=O)CCC(C(=O)N(CCCN(C)C)C)C1C c1(CCCNC(C(C)N(C(=O)CCc2nc[nH]n2)C2CC2)=O)ccccc1 C(=O)(CC(C)C(F)(F)F)NCCC(c1cn(CC(C)NC(C(CCC#C)O)=O)nn1)CC C(=O)(C(C)C(C)NC(=O)C(C)c1ccco1)NCc1cn(CC)nc1 C(CCCCC(=O)NC(C(=O)N(C)CCc1cccnc1)C1CC1)N(C)C C1(OC)(CNC(C2CC(SC)C2)=O)CCN(C(=O)CSc2nncs2)CC1 N1(C(C23N(C(C(C)Cc4ccccc4)=O)CCC2C3)=O)CC2(CCNC(=O)O2)C1 C1(NC(C(c2cnn(C)c2)NC(C(C)c2cccs2)=O)=O)CCCC(O)C1O C=CC(C(=O)N(C)CCOCCNC(c1n[nH]cc1F)=O)c1ccccc1 c1(C(N2CCC(C(=O)NC(CC#C)C(N)=O)CC2)=O)ccc(C=C)cc1 C1(NC(CC=CCC)=O)CN(C(=O)CC(C)F)C2(CCCCCC2)C1 N1(C(c2c(C)cco2)=O)CCC2CCN(C(=O)CCCc3cccnc3)CC2C1 OC1(CNCc2cn(-c3ncccc3Br)nn2)CCc2ccccc21 C12(C(=O)OCC(c3ccco3)OC)CN(C(=O)OC(C)(C)C)CC1CCO2.OCO c1(CC)cc(OCC(=O)NC2(C)CCN(C(=O)CC=C(C)C)C2)ccc1Cl CC1C(=O)CCC1CC(N1CCC(C2CCCN2C(c2ccn(C)c2)=O)CC1)=O Cc1ccc(SC(C)C(=O)NCCC2CCN(C(c3ns[nH]c3=O)=O)CC2)cc1 Cc1nc(C)c(CC(=O)NCC2C=CC(NC(=O)Cc3cncc(F)c3)C2)s1 c1(C(=O)NCC(CC)(C)NC(=O)C(C)n2cccc2)cc2c([nH]1)CCCC2 C(=O)(N1CC2COCC2O1)C1N(C(CC(C)F)=O)CCCCC1 Cn1cc(NC(=O)CC2CNC(C(F)(F)F)CO2)c(O)nc1=O C(=O)(N=c1ncn(CCO)[nH]1)C1CC(c2cc(OC)c(C)cc2)(C(=O)O)C1 c1(C(N2CC(CC#N)N(C(=O)Cn3ccnc3)CC2)=O)ccc([Si](C)(C)C)cc1 N1(C(C(=O)Nc2nc(CC)c(CCCC(F)F)s2)=O)CC2CC(C1)C2(F)F c1(C(=O)NC(C2CCN(C(CC(n3c(CC)ncc3)C)=O)C2)C)cc(C)c(C)[nH]1 C1(NC(c2c(OC)cccc2)=O)C2CC1CN(C(=O)CC1(C)CCOCC1)C2 c1(C(=O)NC2CN(Cc3cc(C#N)sc3)CC2O)ccnc2c1OCO2 c1(C(N2CCC3CCN(C(C(C4CC4)OC)=O)C3C2)=O)cc2ncccc2cc1Cl N1(C(c2c(OC)noc2C)=O)C(C)C2CC1C2NC(c1c[nH]c(Br)c1)=O C1(C(N2C(CN(C(=O)CS(C)(=O)=O)C)CCCC2)=O)CC(C)(C)CC(C)(C)C1 C1(C(=O)NCCOCC(N2C(C)(COC)CCC2)=O)CC2CC1CC2O N1(C(CCC=CC)=O)CCC(CCF)(C(=O)O)C1 C(C(C(=O)N1CC(NC(N)=O)C1)C(C)C)NC(c1c(C)cc(F)s1)=O C(CN=c1[nH]c(=NC2COC(C)(C)C2)c2ccc(C)cc2[nH]1)c1cc(C)ncc1 C1(CNC(C(C)CO)=O)CCC2(CCC2)C1NC(c1ccc2occc2n1)=O C1(C(=O)OC)CC2CCC1N(C(=O)C1CC1)C2.N1C(=S)NCC1.C(C)(C)(C)N C1(CC(=O)OCC)CCCCN1C(=O)Cn1cncn1.C1(=O)C(Cn2cncn2)N1 c1(C(N2CC(NC(=O)Cc3cnns3)C(CO)CC2)=O)nc2cnccc2s1 c1(C(N(CC(=O)OC)C(C)C)=O)cc(-n2ccnc2)co1 CCC(CCC(=O)N1C(C)CCCC1C)NC(c1ccncc1)=O C1(CC(=O)NCCCOCCNC(c2nc(O)sc2C)=O)(OC)CCOCC1 c1(CC)c(C(=O)NC(CNC(c2cocn2)=O)CO)cccc1C C(=O)(CC(C(CC)CC)C(CSCCC)=O)NCCOCCCNNC(=O)C1CC1 C1(CNC(C(C)OCCN(C)C)=O)CCCCCN1C(=O)CN1CC=CC1 C1(CC(=O)N(C(CC)C)CC)CC(C)(C)CN1C(=O)CC1CNC(=O)O1 C1(N(C(CSC)=O)C)CCCCC1N(C(=O)C(C)N(C(c1ccccc1)=O)CC)C C1(CCOC)CN(C(=O)C(OC)OC)CCN1C(c1nc(=N)cc[nH]1)=O C1(C(=O)NCc2cn(C3CN(C(c4ccno4)=O)C3)nn2)CC2CCC1O2 CC1(C)COCC1CC(=O)NCCCCCNC(c1snc(O)c1Cl)=O C1(OC)CC2CC(OC)C2C1.N12CC3(CC1CO3)CNC(=O)C1(COC)CC2C1 c1(C(=O)NC(C2(C(=O)NC(c3nccn3C)C)CC2)C)cc(C(N)=O)co1 N1(Cc2c(I)ccc(C)c2)CCc2cc(-c3ccnc(C)c3)ccc2C1 c1(C(N(CCN2C(C)CC2)C)=O)csc(CNC(=O)OC(C)(C)C)n1 N1(C(c2c(C)noc2C)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC1C1CC1 c1(OC)ccc(-n2cnnn2)c(C)c1.N1C(NCC2CC2)=NCCN1C1CCOC1 N1(C(c2c(=N)[nH][nH]c2)=O)CCC2(CCC2)C(NC(C2CCCC(F)(F)C2)=O)C1 c1(C(=O)NCC2=CCN(C(c3c(C)nc(N)cn3)=O)CC2)cccc2nn[nH]c12 N1(C(CC(=C)C)=O)CCCC2CN(C(C3(OCC)CCSCC3)=O)CCC12 Cc1cnnc(O)c1C(N1CC2(NC(C3CCCN3C3CC3)=O)CC1C2)=O C1(COC)C=CCCN1C(C1(NC(=O)CCNC(=O)COC)CC1C)=O S(=O)(=O)(c1cc(C2OCCO2)ccc1C)N(C)CC1CN(CC)C1 CC(C(=O)NCC1CC1C(=O)NCCCc1ccccc1)C(F)(F)F c1(CC)ccc(C(=O)NC2CC(C)N(C(=O)CCC(C)CN(C)C)C2)c(C)c1 NC(=O)CCCCC(=O)NC(Cc1ccco1)C(=O)NCC(=O)NCC1CC1 CCC(C(=O)NC(C(=O)NC(C)CCN(C)C)C(C)CC)C(C)(C)CC CC(C)(C(=O)NCC(CNC(=O)CC1CC2CC2C1)CO)C1=CCSCC1 N1(C(COCC=C)=O)CC(CNC(=O)C(C=C)c2ccccc2)CC1(C)C C1(O)(C(C)C)CCCN(C(=O)CC2COCCN2C(c2ccncc2N)=O)C1 CCC(CC(=O)NCCC(O)C(C)C)NC(c1ccn(CCF)n1)=O c1(C(=O)OC)ccc(C(=O)NCCCCCNC(=O)C(=O)NCCNC(C)=O)s1 C(CC1=CCN(C(=O)CC2(O)CCCCC2)CC1)NC(CC(C)(O)C1CC1)=O C1(NC(C(F)=CCC)=O)CCCC(N(C)C(c2ccc(CF)cc2)=O)C1 CC1(C)CCc2cc(C#N)c(N3CCC(NC(=O)C(F)(F)C4CC4)C3)nc2C1 Cc1sc(C(=O)NC(CNC(c2cc3occc3s2)=O)C2CCC2)c(C)c1C CN1CCCC1C(=O)NCCOCCNC(C1CC1(F)Cl)=O C12CCCN(C1)CCCNC2=O.c1(CNC(C2CC2C2CC2)=O)cccnc1 C1(C(=O)NCCC2CC2)(CC)CCCN1C(c1cn(C)nc1C)=O C(C)(C)(CC(F)C(=O)NCCC1CC(C)C1)NC(C(COC)C)=O C1(c2cn(CCCC(C)(F)CNC(c3c(C)nns3)=O)nn2)CCCNC1=O N1(C(c2ccc(C)c(CO)c2)=O)CCC(C)(C)C(NC(c2ccccc2O)=O)C1 N1(C(=O)NCCCCl)CCCC2CCCCC12.C12CCN(CC1)C2=O N1(C(C=C(CC)CC)=O)CC2CCN(C(c3ccc(C4CC4)s3)=O)CC2C1 n1(CC(=O)NCCN2CCN(C(C(COC)(C)C)=O)CC2)nnc2c1CCCC2 Cc1ccc(C(N2CCN(C(C3(C)CCC(=O)N(C)C3)=O)CC2C)=O)c(N)c1C N1(C(C2CCC(C)(C)C2)=O)CCOC(C)(CNC(=O)Cc2csnn2)C1 C1(NC(C2CC23CCC3)=O)CCC(O)CN(C(c2cccc(Cl)c2F)=O)C1 c1(N(CC(=O)NCC(=O)NCCC2(OC)CN(C(C)=O)C2)C)ccc(Cl)cn1 N1(C(CCS(N)(=O)=O)=O)CC2CCN(C(c3cnc4[nH]ncc4c3)=O)CC12 C1(C(=O)NC(CC(=O)NCCc2c(C)cncc2)C2CC2)CCOC(=O)CC1 CCC(C)(COC)C(=O)NC1CC1NC(c1nccn1C)=O Cc1cccc(C)c1CSC1CCOC1.C1(C2CCOC2)C(=O)N1C1CC1 N1(C(c2c(C)cns2)=O)CC(C)CCC1C(=O)Nc1cccc(CCF)c1 c1(C(C(=O)NCC(=C)C)N(C)CC2CSC2)cnn2c1CCC2 c1(OC)ccc(CC(=O)NC2CCN(C(=O)CCCCC3CC3)C2(C)C)cc1F c1(C(=O)NCC2(NC(C3OCCN(CC)C3)=O)CCCCC2)occ2c1CCC2 Cc1cc(C(=O)NC2CC(O)CN(C(c3ccnc(C4CC4)n3)=O)C2)cc(C)n1 Cc1cc(C(=O)NC2CCN(C(C3CCC3)=O)CC2CO)c(N)c(Cl)n1 N1(CC(=O)N(C2CCN(CC(=O)C3CC3)CC2)CC)CCC(C)(C#N)C1 C(N=c1cc(C(C)(F)F)nc[nH]1)C1CC1NCc1cn(C(c2ccc(Cl)cc2)C)nn1 c1(NC(C2C(CC(=O)NC(COCC)C)CCCC2)=O)ccc(F)c(C)c1 C1(NC(C2C(CNC(=O)CC3CCCSC3)CCC2)=O)CCn2cncc2C1 CC1=C(C(=O)NCC2CC(C)N(C(c3cnccn3)=O)C2)CCCC1 O=C1Cc2cc(CC(=O)Nc3ccc(N4CCC(O)CC4)cc3)ccc2N1 C12(CNC(CC3(C)CC3)=O)CCC(CC1)N(C(c1cn(C3CCOC3)nn1)=O)C2 CC1=C(C)CC(C)(C(=O)NCC2CN(C(C3CCCCC(=O)N3)=O)CCO2)CC1 C1(CC=C)(NC(c2ccc(OCC)cc2C)=O)CCCN(C(c2cn[nH]c2)=O)C1 Cc1nn(C)c(Cl)c1CC1(CC(=O)NCc2cccc(OCCO)c2)CCC1 C(=O)(CS(=O)(=O)CC(C)C)N(CC(C)NC(C1CCC(C)=C(C)C1)=O)CC N1(C(CCc2n[nH]c(=N)s2)=O)CCCCC(CNC(=O)C(c2ccccc2)O)C1 c1(-c2ncn(C(C)(C)C)n2)noc(C2CCCn3cnnc32)n1 Cc1c(C(=O)NC(C)C(C)n2cncn2)cnc(F)c1Br C(=O)(C(O)C(C)(C)C)NC(CCOC)CNC(C1CCCOCC1)=O N1(C(CC)=O)CC2CS(=O)(=O)CC2(CN(C2CCC2)C(C2CC2F)=O)C1 c1(C(N2CC(NC(=O)C(O)c3ccco3)C3(C2)CC3)=O)cccc2nc(O)[nH]c12 C1(C(=O)NCCCNC(c2ccnc(N3CCCC3)c2)=O)CCN(C2CC2)C1=O C1(O)(CNC(C2C(CC(C)(C)C)C2)=O)CN(C(C2CC3CC3C2)=O)C1 C1(CNC(C(CC)COC)=O)C(O)C(O)CN1C(=O)CCC1CCCO1 n1(CC(=O)NC2(CNC(c3cc(Br)co3)=O)CCCC2)cc(Cl)cn1 c1(C(=O)NCC2CC(NC(CC(CC)C)=O)C2)cccc2[nH]c(=N)oc12 C(=O)(C1=CCC(C)(C)CC1)N(C)CCOCCC(=O)N(C1CC=CC1)C c1(C(=O)NCC(C2CCCCC2)C)cc(C2CC2)nn1-c1ccc(Br)cc1 Cc1c[nH]c2cc(C(=O)NC3CCN(Cc4c(F)cccc4I)CC3F)ccc12 C1(C(N(C2CCCN(C(C(F)=C(C)C)=O)C2)CCO)=O)CCc2c[nH]nc2C1 C12(O)CCN(C1)C(C1C3CC4C(C3)C14)C(=O)NC2.CC(C)(C)CCN1CCNCC1 c1(C(=O)NCC(N2C(CNC(=O)CC3CCOC3)CC2)=O)c[nH]nc1[N+](=O)[O-] CCCCCCCCCC(=O)NC12CC1CN(C(C1CN=C3N=CNN3C1)=O)C2 C12(CNC(C(CC)n3ccnc3)=O)CC(CO1)N(C(c1c[nH]c(=NC)o1)=O)C2 CC1CCC=C1C(=O)NC1CN(C(c2cc(Br)nn2C)=O)CC1O C1(NC(c2c(C)coc2C2CC2)=O)CN(C(C2CC23CC3)=O)C2(CCCCC2)C1 CC(C)(C(=O)N1CC2CC2(CNC(c2c[nH]nc2C(F)(F)F)=O)C1)C(N)=O C1(C)(NC(COCC#C)=O)CCN(C(C2CC2c2ccccc2)=O)C1 C=CC(CCC)CC(=O)NC(CNC(=O)C=Cc1cn(C)cn1)CC(C)C c1(OC)ccc2cc(C(=O)NC(C)CNC(c3cccc(F)c3)=O)c(=O)oc2c1 c1(CNC(=O)Nc2c(C)nn(-c3ccncc3)c2)cccc(Cl)c1Cl c1(NCC(CC)(C)CO)ncnc(N2CCN(C34CCC(CC3)C4)CC2)c1C C1(NC(=O)CCN(C(=O)C=CCO)C)CCC(NC)C1.C(=O)(C(C)N)OCC c1(C(=O)NCC2(CCNC(C3C(C)OCC3)=O)CC2)ncn2ccccc12 c1(C(N2C(c3c[nH]nn3)C(C)CC2)=O)ccc(-c2nn[nH]n2)cc1[N+](=O)[O-].CO Nc1ccnc(C(=O)NC2CCN(C(C3CCC(=O)NC3)=O)CC2CO)c1Cl Cc1ccc(C(=O)NCC2C3CN(C(c4nc(Cl)cs4)=O)CC23)c(F)c1F Cc1ccc(N2CCCC2NC(=O)C(=O)N(C)Cc2ccc(C)cc2)cc1 N1(C(c2cc(CC)on2)=O)CCCN(C(=O)CN2CCCC2CO)CCC1 C(=O)(CCC(C(N)=O)NC(=O)NCc1ccc(Cl)cn1)OC(C)(C)C C1(C(=O)NCCC2(O)CN(C(c3cnc(C)nc3C)=O)C2)C2CCC(C2)S1(=O)=O c1(NC(c2c(C(C)=O)ccc(OC)c2)=O)cccc(S(C)=O)c1 C1(O)(C(=O)NC(CC(=O)OCC)C)CC2(CCC(C(=O)OC(C)(C)C)CC2)C1 C1(C(N2CCC(C(N)=O)(NC(c3ccc(C4CC4)o3)=O)C2)=O)CCCCC(=O)N1 c1(C(=O)NCCC2CCC(NC(CS(N)(=O)=O)=O)C2)cnc2c(c1)NC(=O)CN2 C(=O)(CCCCCCNC(c1sccc1CO)=O)NC(C)(C)C(O)CO n1(CC(=O)NCCC2CCC(NC(C3(CC)CC3)=O)C2)ccc2cc(F)ccc12 C1(C(N(CCCC)CCCC)=O)C=CCN1C(C1C=CCS1)=O C1(C)(CN2CC(C)N(c3ccccc3)CC2)Cc2ccccc2C1 c1(C(=O)OC)c(NC(C2CC(F)CN(Cc3ccc(=O)oc3)C2)=O)cccc1Cl C(=O)(CC1=CCCCC1)N1C(C2(NC(C(c3cccc(C)c3)C)=O)CC2)CCC1 c1(CNC(=O)C(c2ccccc2)F)ccc(N2CCN(C(=O)CO)CC2)cc1Cl C12(CNC(=O)COCCc3cccs3)CCC(CN1C(=O)CSC(F)(F)F)C2 O=C1Cc2cc(C(N3CC4CC3CN4C(C3CC3(Cl)Cl)=O)=O)ccc2N1 c1(C(=O)NCC(N(C(C(C)OCCC=C)=O)C)C2CC2)ccc(F)c2occc12 Cc1ccc2c(C(N3CC4CN(C(=O)CC5CCN(C)C5)CCC34)=O)onc2c1 C1(NC(c2ccc(CSCC)cc2)=O)CCCN(C(c2conc2C)=O)CC1F N1(C(C(c2cccc(C)c2)C)=O)CC2CCC1C(NC(=O)C(O)C1CC1)C2 CCCCCC(O)CC(=O)NCC1(C)CCN(C(C2(C)CCC(F)(F)C2)=O)CC1 c1(OCOC)ccc(F)cc1-c1nc(C(=O)Nc2cc(C(C)C)no2)cs1 C(=O)(CC(F)(F)CC(=O)OC)N1CCCN(C(CCCCCCC)=O)CC1.C1CC1 C1(NC(C=CCC)=O)CCCN(C(c2cncn2C)=O)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1CCN(C(C2N=C(C)SC2)=O)CC1C c1(C(=O)NC(CC#C)C(=O)NC(C)COC)cccc2ccoc12 Cc1ccc2c(c1)SC(C(=O)NCC1(F)CC(NC(C3CCCOCC3)=O)C1)C2 C1(C(=O)NCc2ccc(N3CCCCCC3)cc2)CC(O)C(O)CO1 c1(C(=O)NC2CCC2)cccnc1CNC(C1CCCCC1F)=O CCC(C)(C(=O)NC1CN(C(=O)COCC2CCCC2)C1)OC C1(C(N(C2CC(C(=O)OC)C2)C)=O)CC2CCN(C(C34CCC(CC3F)C4)=O)CC12 c1(C(=O)NCCC(C)NC(CCN(C(CC)CC)C)=O)ccc2c(c1)CNC2=O c1(C(N2CC(NC(CCCOC)=O)C(F)(F)C2)=O)cc([N+](=O)[O-])c(F)cc1F c1(CNC(c2c(C#N)nccc2)=O)c(Cl)ccc(F)c1F C1(CNC(c2c(C)nsc2)=O)CC2(CCC2)CN1C(c1ccc(F)c(N)c1F)=O C=C(C)C1OCCC1C(N1CCC(CO)(NC(c2cncc(CC)c2)=O)C1)=O CC1=CC(C)=NS(=O)(=O)N1CC(=O)NCC(O)CNC(=O)C(C#N)C(C)(C)C c1(Nc2cc(C(=O)NC3C(NC(C(C)SCC)=O)C3)ncn2)c(Cl)cccc1Cl n1(CC(=O)NCC(CNC(=O)C(C)(C)CCOC)OC)nc(Cl)ccc1=O c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccc(F)cc1OC N1(C(C(C)=C(C)C)=O)CCC(NC(=O)C(c2ccc(F)cc2)F)CC1C N1(C(C=C2CCN(C)C2)=O)CCOC2(C1)CN(C(=O)CC1CC=CCC1)C2 N#Cc1c(N2CCC(CCNC(=O)CC3CCOCC3)C2)cccc1F N1(C(CNC(CCC)=O)=O)CCCC1CN(C)C(C1(SC2CC2)CCC1)=O Cc1ccnc(C)c1C(=O)NCC1CCCC(NC(C2CC2c2cn[nH]c2)=O)C1 C(C(O)CC(F)(F)F)Oc1cccc(NC(=O)NC2CCCC(OC)C2)c1 N1(C(c2c(C)con2)=O)CCCC2C1CCCCN2C(=O)Cc1ncncc1Cl C(=O)(N=c1[nH]n(C)cc1Br)NCC(CO)OCC Cc1csc2c(C(=O)NC3CCCC3NC(C3(C)CCCCC3C)=O)ncnc12 N1(C(C2C(CC)CN(C(=O)C=Cc3ccoc3)C2)=O)CCCSCC1C c1(C(=O)NCCC(CNC(c2csc(Cl)c2)=O)O)c[nH]c(=O)c2ccncc12 C1(C(=O)NCC(CC(C)C)NC(=O)CCc2cncnc2)CN2CCC1CC2 C1(NC(C(C)c2ccsc2)=O)CC2(C1)CC(CNC(=O)C=CCO)C2 S(=O)(=O)(c1ccc(C)c(C)c1)NC(C(=O)NC(CC)CCCO)C C(c1cc(F)cc(OC(F)(F)F)c1)=CC(CC(C(F)(F)F)n1cncn1)=O c1(OC)cncc(Br)c1C(=O)NCC(O)CN(C(=O)CCC(=O)N(C)C)C C#CC1CN(C(C2(C(C)C)CCN(C(=O)Cc3cnn(C)c3C)C2)=O)CCN1C C1(=O)CCCC(=O)N2CCCC(CC2)N1.C(=O)(C(C)(C)C)N(C)C C1(CNC(c2c(OC)csc2)=O)CC(NC(=O)C=C(C)C)C1(C)C Cc1ccc(C)c(C(N2CC(CNC(c3csc(Cl)c3)=O)CCC2C)=O)n1 c1(C2C(C(=O)NCCN(C(C3C(C)CCC3)=O)C)C2)ccc(Br)c(Cl)c1 C1(NC(CC(C)SC)=O)CC2(C1)CC(NC(=O)Cc1c(Cl)cccc1Cl)C2 C1(CCC)CCCN(C(C2CCC(NC(=O)C(C)N3CCCC3)C2)=O)C1 c1(C(N(CC(COC)C)C)=O)ccc(CNC(c2cc(CCO)on2)=O)o1 N1(C(c2nc(C)oc2)=O)CCC2C(NC(c3cccc(F)c3)=O)C2CC1 c1(C(N2CCC(NC(C3C(C)C3C)=O)C2)=O)cc(Cl)c(Cl)cc1N N1(C(C(C)C)=O)CCCC1C(=O)NCCC1(CO)CC1.c1(C(=O)N)ncc(C(F)F)s1 N1(C(C)=O)CC(O)CC1C(N1CC2(NC(=O)C(c3ccccc3)SC)CC1C2)=O C1(C(C)C)CN(C(C2(F)CC2)=O)CCN1C(c1cc(O)nc(O)n1)=O Cc1nn(C)c(CN(C)CC2(O)CCSC2)c1Cl N1(C(c2cc(OC)c(Br)s2)=O)CCC(C)(c2cn(-c3cncc(Br)c3)nn2)CC1 c1(CNC(=O)NC2CCOCC2)cn(CC2(N3CCCC3)CC(O)C2)nn1 CC(Cc1ccccn1)C(=O)N1CCCC1NC(=O)OCC12CNCC1C2 N1(C(C(C=CCCC)O)=O)C2CCC1CN(C(c1cccc(CC#N)c1)=O)C2 C(CNC(C1CCOC1C)=O)(C(=O)NCCNC(=O)C1CC1)OC C1(C(=O)NC2C(OC)CN(C(c3cc[nH]n3)=O)C2)CC(=O)NC(=O)N1 C(=O)(C1CCc2c(Cl)cccc21)N1CC(O)(CNC(C(C(C)(C)F)(C)F)=O)C1 c1(CC(=O)NC2(CNC(=O)C=CC(=O)NC3CCOC3)CC2)cccnc1Cl C1(F)(C(=O)NC2CCN(C(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)C1 C1(CNC(CC(C)SC)=O)CC(C)(C)CN1C(c1coc(N(C)C)n1)=O C1(CC(=O)NCCOC2CCN(C(=O)CC3CC3)C2)CCCOCC1 C(C(=O)N1CC=CC(NC(=O)C(C)NC2(CO)CCCC2)C1)(C(C)(C)C)OC N1(C(c2ncn(CC)c2)=O)CCC2CN(C(=O)CCC(CF)CF)CCC12 N1(C(CCN(CCCO)C(c2cc(C(C)C)on2)=O)=O)CCCOC(CCO)C1 C1(C2N(C(C(F)=CC)=O)CCC2)CCCN(C(c2ccn(C3CCCC3)n2)=O)C1 Cn1ccn2ncc(C(=O)NCC(C)(C)CNC(c3cccc4c3CCO4)=O)c12 c1(C(C)NC(c2cc(OCC)ns2)C)coc2ccccc12 C(=O)(C1=CC2CC=CCC12)NCC1(NC(c2c(CCC)nco2)=O)CC1 c1(OC)cc(C(=O)NC2CC(F)CN(C(=O)CCOC(C)=O)C2)c(Cl)cc1Cl CC1CN(C(c2ccnc(S)c2)=O)CCC1N(C)C(c1cc(C(C)(C)C)no1)=O N#CCCCCCC(=O)NCC1CCCN1C(=O)C=Cc1ccc([N+](=O)[O-])s1 c1(C(=O)NC2C(NC(C3N(C(C)C)C(=O)CC3)=O)CCC2)ccccc1[N+](=O)[O-] C1(C(=O)NC(CC)C)COC(CNC(=O)C(C)CC2CCCC2)C1 C(=O)(CCCCC(F)F)N1C2CC(CNC(=O)C3=CCCCO3)(OC2)C1 Cc1ccc(C(N2CCC(C)(NC(c3cccc(O)c3C)=O)C2)=O)cc1C N1(c2snc(SC)n2)CCOCC12COCCN(C(c1cc[nH]n1)=O)C2 CC(C)C(C#N)C(=O)N1CCC(CNC(=O)Cc2nn(C)cc2Cl)CC1C c1(C(=O)NC(CN(C(c2cc(C(C)C)ccc2F)=O)CC)C)cnc(N)c(N)c1 C=CC(CC)CC(=O)NC1CCN(C(c2ncsc2C)=O)CC1CC N1(c2cc(N(C)CC3CC=CCC3)nc(COC)n2)CCCC2(C1)CC2(F)F C(=O)(C(C(=O)NCC1CCCC1C(=O)NC1CC2CC2C1)OC)OC N1(C(CCCn2c(C)ncc2)=O)CCN(C(=O)CC2(C(F)(F)F)CC2)C(C)C1C S(=O)(=O)(c1cccnc1)N1CCC(C(C)C(=O)N2CCC2C)CC1 CC(C(=O)NC(CCF)C(=O)NC(CCO)C1CCCC1)C(F)(F)F N1(C(C2CC(OC)C2)=O)CC2(CC1CNC(c1c(C)noc1C)=O)CC2(F)F C1(NC(c2csc(C3CC3)c2)=O)CCCN(C(=O)NC2CC3(CC3)C2)C1 N12CC3CN(CC3C1)C(=O)CCC(C)(C)OC2=O.Cc1ccc(SC(C)(C)C)o1 CC#CCCC(=O)N(CCNC(=O)Cc1cc(C)sc1C)Cc1ccccc1 N1(C(CNc2n(C)c(O)nc2)=O)CC2CC(NC(C3CC4COCC4C3)=O)C1C2 Cc1nn(C)cc1C1=NOC(C(=O)NC2CCN(C(=O)Cn3cccc3)CC2)C1 c1(C(=O)NC2C(NC(CN(C3CC3)CC)=O)COCC2)ccc2c(c1)CC(C)O2 Cc1oc(C2(C(=O)O)CC2)nc1CN1CCC(C2CCCCN2)C1 C=CC1CN(C(=O)CN(C)CCC)CC1NC(c1ccc(-n2cccn2)nc1)=O C1(CC=C)(NC(=O)CC2(NC(C)=O)CC2)CN(C(=O)C(CC)n2cncn2)C1 C1(CNC(C2CC2(Cl)Cl)=O)CCN(C(c2csc3nnsc23)=O)C12CC2 CCC(C(=O)N(C1CC(NC(C2(O)CCOC2)=O)C1)C)n1ccc(C2CC2)n1 C(CC(F)F)(C(=O)NC(C)CCCCCO)N(C(C(CC)C)=O)C C12(CNC(CCCC(N)=O)=O)CN(C(c3ccc4cnoc4c3)=O)CC1CCO2 C1(NC(C2(F)C(C)C2)=O)CCN(C(c2coc3c(Cl)cccc23)=O)CC(C)(C)C1 C1(NC(CCCCNC(N)=O)=O)CCN(C(=O)Cn2cc(C(C)O)nn2)CC1F C1(NC(C(C)CN2CCOCC2)=O)CC2CC1CN(C(=O)Cc1cccnc1)C2 c1(CCC(=O)NCC(C)NC(C2CC3CCC3C2)=O)ccc(Cl)cc1F C1(OC(C2CCN(C(=O)NCC(F)(F)F)C2)=O)C2CCN1CC2 C(C(C(C)C)NC(=O)COCCF)OC.C(=O)(C(C)=C(C)CC)NC(=O)CN c1(NC)ccc(C(=O)NCC(C)(CNC(C2CC(n3cccn3)C2)=O)OC)nc1 CCCCCCCC(=O)N1CCCCC(NC(=O)CN2CCOCC2)CC1 c12ccccc1C2.c1(SCC(N2C(C(=O)NCC(N)=O)CC2)=O)nnnn1C1CC1 C1(NC(c2c(C)scn2)=O)CCCC(NC(C2(C)CCNC2=O)=O)C1 c1(C(=O)NC2(C)CCN(C(C3N(C(C)=O)CCC3)=O)C2)c[nH]nc1S(N)(=O)=O c1(C(=O)NCC(C)(C2CC2)NC(C2N(CC)CCC2)=O)cc(N)c(F)cn1 C(N=c1[nH]c(Cl)ncc1F)C1CN(C(C(COC)OC)=O)C1.CC(F)(F)F C(=O)(CC(C(F)(F)F)NC(c1c(F)ccc(F)c1N)=O)NC1C(C)(C)C(F)(F)C1 c1(C(=O)NCC2N(C(CN(CCC)C)=O)CC(OC)C2)cnn2ncccc12 C(=O)(C(O)CCN(C)C)NC(CC)CN(C(=O)CCc1ccncc1)C C1(O)(c2cn(CC(=C)CC)nn2)CCN(C(C2COC(C)(C)C2)=O)CC1 c1(C(=O)NCC2CN(C(C(C)SC)=O)CC(C)(C)C2)ccc(S(C)(=O)=O)cc1Cl C1(NC(c2cc(OC)ncc2F)=O)COC2(C1)CN(C(c1ccc[nH]1)=O)C2 N1(C(C(C)SCC)=O)CC2C(NC(c3ccc(OCCO)cc3)=O)C2C1 c1(C(=O)NCC2C(NC(c3c(C)onc3)=O)CCC2)c(C)nc2ccnn2c1C C(=O)(CCC(C)(C)C)N(C1CCCN(C(=O)CN2CCCNS2(=O)=O)CC1)C Cc1ccc(NC(C2CC23CN(C(c2cccc(C(=O)OC(C)C)c2)=O)C3)=O)nc1 c1(OC)cccc(CC(C2CC2)NC(=O)C(c2ccc(Cl)nc2)(C)C)c1 C1(c2cccc(C(F)(F)F)c2)(N(C(=O)OCC(F)(F)F)C2CC2)CCOCC1 CCC(CNC(=O)C(C)CNC(C1OCCOC1C)=O)(CC)OC CC1CC(CCNC(c2cc(O)cc(Cl)c2)=O)CCN1C(=O)Cn1cnnn1 N1(CC(COC)O)CCC(N(C(=O)C(C)(C)C2CCOCC2)C)C1 C(=O)(CCCC(C)CCC)N(C1CCN(C(c2c(C#C)cnn2C)=O)C1)CCO O=C1COc2cc(C(N3CC(CO)(NC(c4cnn(CO)c4)=O)C3)=O)cnc2N1 C=CCCC(C(=O)NCC(Cl)=CCl)NC(C1CC(C)CC(=O)N1)=O C1(CN(C(C2CCCOCC2)=O)CC)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(NC(c2nc(COC)oc2)=O)CC2CC1CC2C(N1CCCC(C#N)C1)=O C1(C(N(CCC(=O)NC(c2ccccn2)CC)CC2CC2)=O)CCOC(C)(C)C1 Cc1nn2c(c1CNC(=O)Nc1ccc(-c3ccco3)s1)CNCC2 N1(C(C2OCCN(C)C2)=O)CCN(C(c2c[nH]ccc2=N)=O)C2COCC12 C(=O)(C(c1cccs1)NC(=O)C(=O)NC1CC1)N(CC=C)CC=C C12(CC)CN(C(=O)C(O)CF)C(CNC(=O)COc3ccc(OC)cc3)(C1)C2 N1(C(c2n(CC)ccn2)=O)CCCC1(C)CNC(C1CCOC1C)=O C(C(C)(C)CC(=O)NCCCC1CCCCC1)NC(c1c(OC)cnnc1)=O N1(C(C(CC#CC)NC(=O)C=C(C)C(C)C)=O)CC2CCCC2(CO)C1 C1(NC(Cc2c(C)ccs2)=O)CC(O)CN(C(=O)C(C)(O)c2ccccc2)C1 C(C1=CCCOC1)NCCn1cc(C(C)(C)C(=O)N2CCC(N3CCC3)C2)nn1 c1(SCC(=O)N(C)CC2CCN(C(C(N3CCOCC3)C)=O)C2)ccccc1Cl c1(SCC)cc(CC2CCCC2C(N2CCCC2c2nccc(C)n2)=O)c(C)o1 c1(C(=O)NCC2(CNC(C=CCOCCOC)=O)CC2)ccc[nH]1 N1(C(CCC)=O)CC(NC(=O)C(C)NC(=O)Cc2ccccc2)CC(C)(C)C1 CC1C(C)N(C(=O)CCP(C)(C)=O)CCN1C(=O)CCc1nc(=N)[nH][nH]1 CCC(C)(C)C(O)C(=O)N(C1CCN(C(c2nc(C)oc2OC)=O)C1)CCCC c1(C(N2CC(CNC(c3cn(C)nc3Cl)=O)OCC2)=O)coc2cc(O)ccc12 CC1CCCC(C(=O)NCC2(C(N3CCCC(C(N)=O)C3)=O)CCCCC2)C1 N1(C(C2C(CC)OCC2)=O)CCC2(CCCN2c2ncc(F)cn2)C1 c1(OC)ccc(C(=O)O)c(C(F)(F)F)c1.c12ccc(cc1)CC(=O)N1CCC2C1 N1(C(C(C)OC2CCCC2)=O)CCC(CN(C(=O)CC2CCC(=O)N2)C2CC2)CC1 c1(OC(CC)C)cc(C(N2CCC(CNC(C3CCC(C)S3)=O)CC2)=O)ccn1 CC(C)(C(F)(F)F)OCC(=O)NCC1CC1NC(=O)CCc1cccc(Cl)c1 c1(C(N2CC3(CCN(C(C(C)OCC)=O)CC3)C2)=O)ccccc1C#CC1CC1 CC(C)CC(CC(C)C)C(=O)NCC1C2CN(C(=O)C(O)CC3CCCC3)CC12 N1(C(c2ccc(C)nn2)=O)CCCCCC1CNC(c1cc(C)cc(Cl)c1)=O Cc1cc(CN(c2ccccc2)CC(=O)NC2COC2)cnc1O C1(CNC(C2C(C(=O)OC)CC2)=O)(NC(C2CCCCO2)=O)CCCCCC1 C1(CC=C)CCN(C(C2CCCC2NC(=O)CC2(CC)CCC2)=O)C1 c1(C(=O)NC2CN(C(C3CCCCO3)=O)CC2O)cc2ccccn2c1 c1(CC)cncc(C(=O)NC(CNC(c2cnn(C)c2)=O)(CC)CC)c1 Cc1ncc(CNC(c2cnn(CCNC(c3cnsc3)=O)n2)=O)n1C Cc1cccc(C)c1CC(=O)NCC1CN(C)CCN1C(=O)C(F)C1CCCC1 C1(N(C(=O)C(CC2CCCC2)OC)CC)CCN(C(c2ccc(O)nc2)=O)CC1 C=CC(C(F)(F)F)NC(C1CC(O)CN1C(=O)CCC1CC1(F)F)=O N1(C(C=CC(CC)=CC)=O)CCN(C(c2cc(C)n(C)n2)=O)CC1CC(F)F c1(OC)cc(C)cc(CN2CC(C(=O)Nc3ccnc(F)c3F)C2)c1O Cc1cc(O)ccc1C(=O)NCC1CCN1C(=O)C(F)n1ccnc1 c1(C(N2CC(CNC(C(C(=O)OC)C)=O)C2)=O)csc2ccc(F)cc12 c1(NCC(Cc2cccc(OC)c2)N)nn(C)c2ncc([N+](=O)[O-])cc12 c1(C(=O)NCC(CNC(C(C=C)O)=O)F)sc2cccc(F)c2c1COCC c1(C(N2CC(C)CC(NC(c3c(OC)cccc3)=O)C2)=O)ccc2c[nH]nc2c1 c1(NCC(c2c(Cl)ccc(C)c2)O)ccc(C#N)cc1Cl C(CC)(C(C)(F)F)(c1n(CCCOCC)nnn1)NC1CCCN(C(N)=O)C1 Cc1ccn(C)c(=NC(=O)N2CCC(C3CCCO3)CC2)n1 CC#CCC(C)N=c1ccnc(NCCn2cnc(CO)c2)[nH]1 N1(C(c2c(CCC)n(C)nc2)=O)CCCC(NC(c2occc2C)=O)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)NCC(CC)NC(c1cccc(Cl)c1C)=O N1(C(c2ccc(OC)nc2)=O)CCC(C)C(NC(C2CSC2)=O)C1 C1(CCNC(C(CC2CCCC2)N(CC(=O)OCC)C2CC2)=O)CC2C=CC1C2 C1(NC(C(C)NC(N)=O)=O)CCCCCC1NC(c1nc[nH]c1C(F)(F)F)=O c1(C(=O)NC(CC)(CNC(=O)C=Cc2cccn2C)CC)ccc2ccnn2c1 c1(C(N(CCCSC)Cc2nc[nH]n2)=O)ccc(C)cc1Cl N1(C(C)C)CCC(C(=O)NCC(F)C(=O)OCc2cc(Cl)cn2C)CC1 C1(NC(C2N(C(=O)COC3CC=CC3)CCN(C)C2)=O)CCn2cnnc2C1 C(C(=O)NCCOC1CN(C(=O)C(c2ccccc2)O)C1)(C(C)C)NC(=O)OC CC1CN(C(C2CCC(O)CC2)=O)CC1NC(c1ccc(CC2CCC2)cc1)=O N1(C(CCOCC#C)=O)CCC2(CC1)CC2CNC(=O)C=CC C1C(=O)N=C2C=C(N(C)N2)O1.C1(C(N(CCC)C(C)C)=O)CCN(CC(C)C)C1 c1(N(C(CC2CN(C(C(COC)O)=O)CC2C)=O)C)ccc(C)c(C)c1 C#Cc1cn(C)nc1C(=O)N(CCCCCNC(C1CCCO1)=O)C CC1(O)CCN(CC(N2CC=CC(NC(=O)CCN3CCCS3(=O)=O)C2)=O)C1 N1(C(C(C)Oc2ccccc2)=O)CC(CNC(=O)CNc2nccs2)C(F)(F)C1 CCN(Cc1cccc(Cl)c1)N1CCN(CC(=O)NC)CC1 C1(CNC(C(C)(C)OCC)=O)CCC2CN(C(c3cc(C)ns3)=O)CC12 c1(-c2nc(-c3ccc(OCC)c(OC)c3)nn2CC(N)=O)ccn2ccccc12 C1(CCNC(C(CCCC)C)=O)CCN(C(=O)CNC(=O)C(C)C)CCC1(F)F C1(C(N2C(CNC(=O)Cn3cccn3)CCC2)=O)CC2(C1)CC2F c1(N(C(C(C2CCOC2)OC)=O)CC(C)C)cc(C)ccc1F CC(C)C(CO)ONC(=O)C=CCF.C1(C(=O)N)C(C)C1C c1(CC)c(CN(C(c2cccnc2)C)CC)oc2ccc(Cl)cc12 C1(C(C)(C)F)CCN(C(c2cc(Br)sc2Cl)=O)CC1 N1(C(CCN(C(=O)Cc2nnc(C)o2)CC=C)=O)CCN(C)CC1C C1(C(=O)NCC(CC)(CC)NC(C2SCCS2)=O)CC(C)(C)CN1C CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1ccccc1CC#N)=O Cc1cc(CNC(=O)CC2CCSCC2)oc1C S(=O)(=O)(CC(=O)N(C(CC)C(=O)NCCC(C)CCO)C(C)C)NC C1(C(=O)NCC2CC(NC(C=CC(C)C)=O)CC2O)Cc2c(F)cccc2O1 Cc1nc(C(=O)NCC#CC(=O)N(CCC(C)C)CCO)c(C)s1 N1(C(C=C(C)Cl)=O)CCCC2CN(C(C3COc4ccccc4C3)=O)CC12 C(CC(=O)NCC(CO)C1CCC1)(C(F)F)NC(c1ccc(CC)cn1)=O C1(CC)(Cn2cc(-c3sccc3C)nn2)CC(F)(F)C1.C1C(=O)N1C1CC1 C1(C(=O)NCC(C)NC(=O)C(O)C(C)(C)C)CC2COCC(C1)C2(F)F c1(C(N2CCCC(C3(C)COC(=O)N3)C2)C(=O)NCCOC)cccc(CO)n1 Cn1nnc(=NS(=O)(=O)c2ccc(C(=O)NCCCCNC(=O)C3CC3)cc2)[nH]1 Cc1nsc(C)c1C(N1CCC(CCNC(=O)CC2CCC(C)CC2)CC1)=O C1(CNC(C(C)(C)F)=O)C2CCC(C2)N1C(c1ccc(Cl)c(O)c1)=O C1(C(N2CCC(CN3C(=O)CCCC3)CC2)=O)CCC(C(N)=S)CC1 C1(C(C)NC(=O)CC2CC(=O)C2)CCN(C(C2(CF)CC2)=O)C1 C1(NC(C)CCCCNC(=O)OC(C)(C)C)CCNC(=O)CC1 C1(CC(=O)N(CCCN(C)C(C2CC2c2ccccc2)=O)C)CCCNC(=O)C1 c1(C(N(C)CCc2cn(CCCOCC(F)F)nn2)=O)cnc2scnc2c1 N#Cc1ccc2nc(NC(C3CC(NC(c4cccc(F)n4)=O)C3)=O)[nH]c2c1 C1(NC(Cc2c(C)noc2)=O)CCCN(C(=O)Cn2cnnc2)CC1 C#Cc1ccccc1CNC(=O)C(C)N(C(C1CN2CCN1CC2)=O)C1CC1 C1(NC(CCCC#C)=O)CN(C(C2CCCC(C)(C)O2)=O)CC2(CCOCC2)C1 CC(C)C(C(C)NC(c1cn(-c2ccccc2)nn1)=O)NC(=O)C(N)=O C1(C(=O)NCC)CCCC12CCN(C(=O)NCC13CCCC1(OC)C3)CC2 Cc1nc(CC(=O)NCc2cc(NC(=O)CN3CC4CC4C3)ccn2)c(C)s1 c1(C(=O)NC(CNC(CC(COC)C)=O)C2CCC2)cccc(N)c1O N1(C(CCSCC)=O)CCCC(O)(CNC(C2CC2C)=O)C1 CCCC(C(=O)NC(COC(C)=O)CO)NC(c1nc(O)sc1C)=O N1(C(c2c(C)nco2)=O)CC(NC(c2ncnc(O)c2Cl)=O)CC(C)(C)C1 c1(C(=O)NC2CC(NC(C3(F)CC3Cl)=O)C2)nsc2cc(Br)ccc12 c1(OC(C)C(=O)NCc2cccc3c2NCC3)ccc(Cl)cc1C(F)(F)F C#Cc1cc(F)c(C(N2CCCN(C(C3CCCCS3)=O)CC2)=O)cc1F c1(N(NC)C)cccc(CN2CCOCC2)c1.c12ccsc1Cn1ccnc1-2 C12(NC(CC=C)=O)COCCC1CN(C(=O)CCc1cn(C)nn1)C2 N1(C(C(=O)NCCOCCCC)=O)CCC(C)(NC(=O)C2=COCC2)C1 c1(OC)ncnc(N2CCCC(O)(CNC(c3ccc(Cl)nc3C)=O)C2)c1OC N1(C(C2C(C=C(C)C)C2(C)C)=O)CCN(C(c2ccsc2C)=O)C2(CCC2)C1 N(C(=NCC1CCCN1C(C)=O)NCc1cn(C)cn1)C1CCN(C(CC)=O)C1 C1(NC(C2C(C(C)O)C2)=O)CCC2CC1CN2C(C12CCCC1C2(F)F)=O c1(C(=O)NC2C(NC(=O)C(O)CCCc3ccccc3)C2)nnn2c1CSCC2 C#Cc1ccc(Cl)c(C(=O)NCC(C)NC(=O)C(C)(CO)NC(C)=O)c1 c1(C(=O)NC2CC(NC(CSc3nc(C)[nH]n3)=O)C2)n[nH]c(C)c1F Cc1ncnc2c1CC(C(N1CCN(C(=O)CP(C)(C)=O)C(C(C)C)C1)=O)CC2 N1(Cc2cccc(OC)c2O)CCc2c(C(=O)NCC(C)O)n[nH]c2C1 CN1CCC(C(=O)NCC2CNC(=O)C2)(NC(=O)CS(C)(=O)=O)C1 Cc1ccc(-c2n[nH]c(CN(CCCNC(=O)CC(C)(C)F)C3CC3)n2)cc1 c1(CN2C(CC(=O)Nc3cc(C)c(Br)cc3F)COCC2)ccc(O)c(C#N)c1 c1(C(=O)NC(CCC)CCCNC(=O)CS(N)(=O)=O)cc(F)c(C)cc1F C1(CNC(c2n(C)nc(CNC(=O)C(C)(O)C3CCC3)c2)=O)CCCOC1(C)C CCCC(CCCNC(C1CC(SC)C1)=O)NC(C1OCCN(C)C1=O)=O Cc1cccc(-c2cn(C3CC(C(=O)N(CCCF)C)C3)nn2)c1C(=O)O Cc1cc(F)ncc1C(=O)NCC1CCCN(C(=O)CSS(C)(=O)=O)CC1 N1(C(C2N(CN(C)C)C(=O)CC2)=O)CC2CCN(C(c3cc(Br)n[nH]3)=O)C2C1 CCCC(CC)C(=O)NC(C)(CNC(=O)Cc1cncn1C1CC1)CC N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)Cn2nc(C)cc2C)C1(C)C N1(C(CC)=O)CCCC(C2CN(C(=O)COc3ccc(C)cc3)C2)C1 C1(C(N2CCC(N(C)C(c3cc(C4CC4)no3)=O)C2)=O)OCCC1(C)C c1(C(=O)NC2CC(CNC(CC3CCC(=O)C3)=O)C2)ccc2ncsc2c1 c1(C(=O)NC(CNC(c2n(CC)ccc2)=O)(C)C2CCC2)csc(C)c1C c1(C(=O)NC(C)CN(C)C(C2(C)CCSCC2)=O)cc2cccc(Cl)c2s1 c1(C(N2C(C(C)NC(=O)C=C3CCC3)CCC2)=O)cncc2[nH]ccc12 c1(C(N2CCC(O)(CNC(C34CCCC3OCC4)=O)C2)=O)n[nH]c2c1COCC2 C1(CC)CN(C(=O)C(C)N(C)C)CCN1C(c1ccc(OC(F)(F)F)cc1)=O N1(C(c2c(C)n(C)cc2)=O)CCOC2(C1)CN(C(c1cccc3c1OCC3)=O)C2 CCCCC(CN=c1[nH]ccnc1F)NC(c1ncccc1Cl)=O N1(C(C(CSC)O)=O)CCC2CN(C(c3cncs3)=O)CC2C1 C(C(O)CN=c1nc(C2CCCC2)[nH]s1)NC(C)=O.C1(C)(C)C(=O)N1C1CC1 CC[Si]1(CC)CCN(C(=O)NC(c2cccc(C)n2)C)CC1 c12ccccc1OC(=O)C2.C(=O)(CC(C)(F)F)N1CCC(C(=O)NCCCC)C1 C1(C(C(=O)NC(C)Cc2cnn(C3CCOCC3)c2)F)CCC(=O)CC1 N(C(=NCc1ccnc(OC)c1)NCC1CCCC1)Cc1n(CCOC)nnn1 C1(C(=O)NCc2c(C(N3C(C(=O)NC)C=CC3)=O)n[nH]c2)CCCCCCC1 C1(NC(CNC(N)=O)=O)CN(C(=O)CC2CC3(COC3)C2)CC1S(C)(=O)=O N1(C(C2=NOC(C)(C)C2)=O)CC(NC(C2C3CCCCC23)=O)CC12CCCC2 CC(C)(C)C1=NOC(C(=O)NCC(C2CCCN2C(c2ccc(F)s2)=O)(C)C)C1 N1(C(c2c(F)ccc(C)c2)=O)CCOCC(C)(CNC(C2C3CCOCC23)=O)C1 CCC(CC(=O)NCC(CC(=O)NCC1(CC(=O)OC)CC1)OC)C(C)C n1(CC(=O)N(C(CN(C(CN(CCOC)C)=O)C)C)C)ncc(Cl)c1C c1(CC(=O)NC2(CO)CCN(C(=O)CCc3cccs3)CC2)ccc2c[nH]nc2c1 C1(NC(C(CC#C)O)=O)CCN(C(c2ccc(OC)cc2OC)=O)C12CCC2 CN1CC(C)(C)CC1C(N1CC(O)CC1CNC(C1(CC2CC2)CC1)=O)=O N1(C(CCN(C(CCC)C)C)=O)CCc2sc(CNC(C3CC3C)=O)nc2C1 C1(NC(C(CC)SC)=O)CCC2CN(C(c3cnc(SC)[nH]3)=O)CCC2C1 CC(C)CS(=O)(=O)CC(=O)N(C1CCN(Cc2c[nH]c3cc(F)ccc23)C1)C c1(C(=O)NCC2(NC(C3(C#N)CCCOC3)=O)CC2)[nH]c2ccc(F)cc2c1Cl n1(CC)ncc(C(N2CCCC2C(C)NC(C2(O)CCC2)=O)=O)c1Br c1(C(=O)NCCCOCCN(C)C(C2CCC3(CCC3)C2)=O)cc(F)cc(Cl)c1 c1(C(N(CC(C)CNC(c2cc(N)c(F)cn2)=O)C)=O)cc2ncccn2n1 c1(C(N(C2CCN(C(=O)CCn3ccnn3)C2)CC#C)=O)csc(CO)n1 C12(NC(CCOCCC)=O)CCN(C(c3cncc(OC)c3)=O)CC1C2 c1(C(=O)NC(C)C(C)NC(c2ccc(F)cn2)=O)cc(N)nc(Br)c1 C1(CCCC)CN(C(C2CC(C3CC3)=NO2)=O)CCN1C(c1sc(C)cc1Cl)=O c1cnc(NCCNC2CCCC2O)c2cncn12 C(=O)(CCS(N)(=O)=O)NCC1C(CNC(C2N(C(=O)NC)CCC2)=O)C1 Cc1[nH]c(=N)[nH]c(=NCCc2nc(Cl)cs2)c1[N+](=O)[O-] C(CC(=O)NC1CCC1C1CCC1)(C(F)(F)F)N(C)C C(=O)(C1Cc2ccc(F)cc21)NC1(C)CN(C(=O)C2Cc3cccc(Cl)c32)C1 C1(CC(=O)NC(CC=C)CNC(=O)CN(C)C(N)=O)CCC(C)(C)C1 C(=O)(C1=NOC(C)C1)NCCC(C(C)C)NC(C1N(CC)C(=O)CC1)=O CC(C)CC(CNC(c1cn(CC(F)(F)F)nn1)=O)NC(=O)C(F)C(C)C c1(OCC(=O)NC2CCN(C(CC)=O)CC2O)cc(F)c(F)cc1F C#Cc1cc(C(=O)NC2CCCCC2NC(c2cn(C)nc2C)=O)cc(Cl)c1 N#CCCCCCC(=O)N1Cc2[nH]nc(C(=O)NC3(C4CCCC4)CC3)c2C1 c1(C(=O)NC2CCN(C(Cc3scc(CC)n3)=O)C(C)C2)ccc2ccsc2c1 c1(C(N2CC(N(C(C3C(C=C)OCC3)=O)C)C2)=O)cc(OC)cc(Br)c1N CC1CCN(C(c2cn(C(C)(C)C)nn2)=O)C1CNC(c1nc(C2CC2)cs1)=O CC1(C)OCC2CC12C(N1CCOCC1CCNC(=O)Cc1ccnc(O)c1)=O CC(C)CC(C)C(=O)N1CCCC(CNC(c2ccn(C)c2)=O)C1 c1(C(=O)NCC(O)CNC(C2(N(C)C)CCOCC2)=O)ccnc2ccnn12 C(=O)(CC1=CCN(C)CC1)N1C(C)CCN(C(=O)CC2CCC(=O)N2)CC1 c1(OC)cc(C(=O)N(C)CCNC(C2CSCN2C(=O)C(C)(C)C)=O)ccc1F C1(NC(C2ON=C(C)C2C)=O)CN(C(=O)Cc2c(C)cccc2C)C2(CCC2)C1 C(=O)(C(O)CC(N)=O)NCC1(O)CC(CNC(c2cnn(C)c2C(F)(F)F)=O)C1 C(=O)(C1CCc2cccc(F)c21)NC1(C)CCCN(C(c2c(C)csn2)=O)C1 c1(CC(C)C)nccc(C(=O)NCC2(C)CCN(C(C3(F)CCOC3C)=O)C2)n1 N1(S(CCSc2ccc(F)cc2)(=O)=O)CCN(CCOC)C(C)C1 N1(C(c2n(CC=C)ccc2)=O)CCC2(CCN(C(=O)CN3CCC(C)C3)C2)C1 c1(CCC(=O)OCCCCCF)c(Br)cc(Br)c2cccnc12 C(C(C)(C)CC(=O)NCc1c[nH]c(C)cc1=O)NC(c1c(C)n[nH]c1)=O c1(C(N(C(CNC(CN(CCOC)C)=O)C)C)=O)ccc(F)c(OC)c1F C1(CNC(CC(C)OC)=O)COC(C)(C)CN1C(=O)Cc1cn(C)nc1C C=C(C)C(CC(=O)NC1CCC(N(C)C(C2CCC(C)(C)CC2)=O)CC1)OCC C1(O)(CC#C)CC(C(=O)NC2CC(N(C(=O)Cn3cccn3)C)C2)C1 c1(C(=O)NC2(CNC(CC3C(C)C3)=O)CCC2)ncccc1CO N1(C(C2N(C)C(=O)CC2)=O)CCOCC(C(N2CC=CC2C(=O)O)=O)C1 c1(SCC)ccc(C(N2CCN(c3cccc(O)n3)CC2)=O)c(Cl)c1 c1(CC(N2C(CNC(c3n(CC)nc(C)c3)=O)CC2)=O)ccc2c(cnn2C)c1 CCC(C)C(C)C(=O)N1CCOCC1CN(C(=O)C(F)CC1CCCC1)C N1(C(C(CC=C)C)=O)CCN(C(c2cnc3cc[nH]c3c2)=O)CC(C)C1 Cc1cc(C)c(C(N2CC(NC(=O)CC3CCC(F)(F)C3)C(C)C2)=O)c(O)n1 Cc1ncccc1CNC1CCC(NC(c2sccc2Br)=O)C1 c1(-n2c(C(=O)NCC(CNC(C3CC(C)C3)=O)O)cnc2)cccc(Br)c1 C(C1CCN(C(C2CC3CC3C2)=O)CC1)=CC(=O)N(C1(C)CC1)C c1(SC(C)C)ccc(C=CC(=O)Nc2cc(C(F)(F)F)ccc2C)cc1 n1(CC(=O)N(CCNC(=O)C(C2CCCCC2)F)CC)ncc(Br)c1C C1(CC=C)(NC(=O)C2=C(Cl)CCOC2)CC2CCC(C1)N2c1nc(Cl)ncc1Cl N1(C(c2c(C)cncc2Br)=O)CCC2CN(C(C3CCCCC3O)=O)CC12 c1(C(=O)NCCCNC(=O)CCSCC2CCCC2)ccccc1 CCC(C)C(C(=O)NCC(CO)CC(C)C)N(C(c1cn(C2CC2)nn1)=O)C Cc1cc(F)cnc1C(N1CCC(Cc2cn(Cc3ccccc3Br)nn2)CC1)=O C1(C(N(C2CN(C)C2)C)=O)(CC)CN(C(=O)C(c2ccccc2)O)C1 C1(CNC(C2(SCC)CC2)=O)CN(C(C2CCNC2=O)=O)C2CCCCC12 CN1C(=O)C(=O)N(CC(=O)NCC2C=CC(NC(C3(C)CCCC3)=O)C2)C1=O C(=O)(CCCCC(N)=O)N1CCC(C)(N(CC#N)C(c2ccc(C(C)O)cc2)=O)C1 c1(C(N2CC(NC(=O)C=Cc3cn(C)cn3)CC(C)C2)=O)cc(F)c(Cl)cc1F C1(C(N2CC(CNC(C3(CC=C)CCOCC3)=O)C3C2C3)=O)CCCC2(CC2)C1 Cc1nc2ccccn2c1C(=O)NC1CC(CNC(C2C3CCC(F)(F)C23)=O)C1 CC1C(NC(c2ccnc(Cl)c2)=O)CC2CCC1N2C(c1nc(F)ccc1Cl)=O C1(CC)CC(C(=O)Nc2cnc(C)nc2)CCN1C(C1CCSC1)=O C(C(O)CC1CCCCC1)(OCC)NC(c1cnn(CC)c1)=O N1(C(c2c(C)ccc(O)c2)=O)CCC2CCN(C(C3CCCN(C)C3)=O)C2C1 C1(C(=O)NC(C(N2CCCC(CCF)C2)=O)C2CCOC2)CC2CC1CC2O c1(C(=O)NCCC2CCCN(C(CC3CCC(=O)O3)=O)C2)ccn2nccc2c1 C1(C(N(CCNC(c2cc(CC(C)C)[nH]n2)=O)CC)=O)COC(C)(C)C1 c1(C(N(C(C)C(=O)NCC2CCC2NC)CC)=O)cscc1OC C(=O)(CC(C)CC(C)C)NC1(CNC(C2CCCN(C(CC)=O)C2)=O)CCCC1 c1(C(=O)NCC(CNC(c2ccc[n+]([O-])c2)=O)CO)cccc2c1COCC2 C(CCS(C)(=O)=O)(C(=O)NCC1CCCCN1C(=O)COC1CCOCC1)OC C=CCCCC(C(=O)NCC12CC(CN1C)C2)NC(=O)Cn1ccc(C)n1 C1(N(C(C2C(C)CC2)=O)C)CCC2CN(C(=O)CCOc3cccnc3)CC12.C1(O)CC1 CC1CCN(CCC(=O)NC2CC2NC(=O)CC2CC(=O)NC2=O)CC1 C1(C(=O)NCCCCC(N)=O)CCN(C(=O)CC2(O)CCOC2)C12CC2 C(C(=O)Nc1nc(Cl)ccc1Br)(C1=NOCC1)N1C(CC(=O)NC)CCCC1 N1(S(CC(C)C)(=O)=O)CC(NC(C2CC(=O)N(C)C2)=O)CC2(CCOCC2)C1 N1(C(C2OCCN(C)C2)=O)CC2(CC2)CC1CC(=O)NCCC(N)=O C(=O)(CC(F)(F)CC)NC.C1C(C)NC(=O)C=CCN1CC C1(O)(C(=O)NC(CC(C)NC(C2CCc3nc[nH]c3C2)=O)C)CCCC(C)(C)C1 O=S(=O)(c1ccc2[nH]c(=NCCCCCO)sc2c1)NCCOc1ccncc1 c1(C(=O)NC(C2OCCN(C(C(C(CC)C)C)=O)C2)C)cccc2sccc12 C1(NC(CSCC(=O)OC)=O)CCC(NC(=O)CC2CCC(C)CC2)CC1 c1(CNC(C2(CNC(=O)CCOC3COC3)CC2(F)F)=O)cccnc1OC C1(C(=O)NC(CNC(CCOCCOC)=O)C)CCC2(CC2)C1 N#Cc1cc(C(N2CC(NC(=O)COCC(F)(F)F)C(F)C2)=O)ccc1O N1(C(C(CC#C)C)=O)CCC2(CCCN2C(=O)CN(C)C(C)=O)C1 C1(NC(c2ccc(OCCC#C)cc2)=O)CCN(C(C2(CC)COC2)=O)CC1O N1(C(C=C(C)C2CC2)=O)CCC2(CC(NC(=O)Cc3csc(C4CC4)n3)CO2)C1 c1(C(=O)OC)ccc(O)c(NC(C2CN(C(C3CCCO3)=O)CCC2O)=O)c1 CC1CCCC(CC(=O)Nc2ccccc2C(F)(F)F)O1 CC(C)CC(C(=O)NCc1cnc(=N)[nH]c1)NC(c1nnc(O)nc1O)=O C(=O)(C(C)(C)C(C)(F)F)NC1CC(NC(c2nc(C(C)C)oc2)=O)C12CCC2 C1(COC)(NC(=O)CCC(F)F)CCN(C(=O)C#CC2(C)CC2)CC1 N1(CCNC(=O)CCn2cccn2)CCN(C(C2CCCC(O)C2)=O)CC1 c1(CCNC(=O)NC(c2ccc(F)cc2)C)ccc(OC)c(Cl)c1 N#Cc1ccc(C(=O)NCC2OCCC2C(=O)N(CC(O)CO)CCO)o1 C(=O)(CCCCCC(C)O)NCC(CN(C(C=CC(CC)C)=O)CC)(C)C C1(NC(C(CC)CC)=O)CC(CNC(=O)Cc2cnn(CC)c2)C12CCC2 CC1CC(C(=O)N(CCCn2cc(COCC(N)=O)nn2)C)CO1 c1(C(=O)NCC2(CCNC(C(CSC)C)=O)CC2)ccc2n[nH]cc2n1 c1(C(=O)NC(C)(C)CCNC(C2CCCS2)=O)ccnc(C2CC2)n1 C(CC(=O)N(c1csnc1C)C)(C(F)(F)F)NC(c1cccc(C)c1O)=O N1(C(C2C(C#C)C2)=O)CC(NC(C2(n3cncn3)CC2)=O)CC(F)C1 C1(CC(=O)NC2CN(C(c3cc4n(n3)CCO4)=O)CC2O)SC2=NCCN2C1=O C(CC(C(C)(C)C)NC(=O)C(C)(Cl)Cl)N(C(=O)CCC1CC1(C)C)C c1(OC)cc(C(N2CCC(C)C2CNC(c2csnn2)=O)=O)ccc1F c1(CC)c(C(=O)NC2CCOCC2NC(c2[nH]cnc2C)=O)sc2ccccc12 C1(C(N2CC(C(=O)NCCSCC)C2)=O)CCOC1(C)C c1(SC)ccc(C)c(C(=O)NCC2CC2(C)C(F)F)c1 C1(C(=O)OCC)CCN(c2cc(N3CCCC(c4nnc(C)o4)C3)ncn2)CC1 n1(CC)ccnc1C(=O)NC12CC(C(=O)Nc3cnsc3)(C1)C2 C1(C(=O)NCC2N(C(C(C)=CC)=O)CC2)CCC2(CC2)N1C(=O)OCC.C(C)(C)C N(C(=NCCCOC)NCc1noc(C)n1)CC1CC(OC)C1(C)C NS(=O)(=O)CCC(=O)N1CCCC1CNC(=O)CC1CC(O)C12CCC2 CCC(C)CC(=O)NCc1cn(CC(N2CCC(CC3CCCO3)C2)=O)nn1 C1(C2CC2)(NC(c2noc(CC)c2C)=O)CCN(C(=O)CC2CC2C(F)(F)F)C1 c1(CC)cnccc1C(=O)NC(CCF)C(=O)NCC1CCN(C(N)=O)CC1 C(=O)(C#CC(C)(C)CNC(c1cccn1C)=O)NCc1cc(OC)nn1C C1(C(C)C)CCC(C)CC1C(=O)NC1CC12CC(NC(C1(F)CCCCC1)=O)C2 c1(C(c2nnnn2C(C)(C)C)NC(CC)(C)C)nc2ccc(Br)cc2o1 N1(C(c2c(C(C)C)n[nH]c2)=O)CCCC(C(=O)NC2CC(CCC(N)=O)C2)C1 n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CCCC(F)C2)c(C)n1 C1(NC(CC(CNC(C2(C)CCCCC2)=O)OC)=O)CN(C)C(=O)C12CC2 CCCC#CC(C)(C)NC(C1CCN(C(=O)CC2CC=CC2)CC1O)=O C1(C(N2CCCC2c2cn(Cc3cccc(Br)c3F)nn2)=O)CCCCC12CC2 C(C(=O)NCCCN(CC(N)=O)C)(N(CCCN)C)SCC.CO C1(C)(CNC(Cn2nnc(C)n2)=O)COCCN(C(c2cnc(Cl)cc2N)=O)C1 C#Cc1ccc(C(N2CC(CNC(c3c[nH]nc3-c3cnn(C)c3)=O)C2)=O)nc1 C(=O)(C1Cc2ccccc21)N1C(C)CC(C(N2CC(O)(c3nn[nH]n3)C2)=O)CC1 CCCC(C(O)C(=O)NC(c1ccco1)C)NC(=O)C(C)NC=O Cc1cc(C(=O)NC(CNC(c2cnco2)=O)C(C)C(C)C)cc(C)c1F O=C(C#CC1CC1)NCC1CCCN(C(=O)CCc2ccccc2Br)C1 CC(C)CS(=O)(=O)CC(=O)NC12CCC(CC1)N(C(C1CCOC(CF)C1)=O)C2 C(=O)(CCCCN(C)C)NCCCOCCN(C(CC(C)C)=O)C C1(NC(c2c(Cl)cnc(C)n2)=O)CN(C(C2CC2CC(C)(C)C)=O)C2(CCOC2)C1 C1(NC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)CC2CCCC23CC3)CC1F c1(CN(C(C(CCC)O)=O)C)cnn2c1CN(C(c1sc(OC)nc1Cl)=O)CC2 c1(C(N2CC(NC(C(CCC)NC(N)=O)=O)C3(C2)CC3)=O)ccnc2cc[nH]c12 C1(NC(N(CC)CC)=O)(CSC2CCS(=O)(=O)C2)CCCSC1 C1(C(N(C(CC(C)C)C)C)=O)CCN(C(c2ocnc2C2CC2)=O)C12CCC2 c1(NC(=O)CSCCN(CC=CC#C)C)ccc(OC)cc1 O=C1CCC(CCC(=O)NCC2CN(C(=O)C(F)(F)C3(O)CCC3)CCO2)=NN1 C1(CC(=O)NCCF)CCC2(CC1)CCN(C(=O)C(F)(F)c1ccncc1)CC2 C(CC(=O)N1CCCc2nccn21)=CC1CN(C(C(CCCC)C(C)C)=O)C1 C(=O)(CCS(=O)(=O)N(C)C)N(C1CC1)CC1N(C(CC2CCN(C)C2)=O)CCC1 c1(NC(N2CC(C(=O)Nc3ccc(N(C)C)cc3)C(O)C2)=O)cc(Cl)ccc1Cl N1(C(C(C)=C(CC)C)=O)CCCC(N(CCF)C(c2cc(COC)oc2C)=O)C1 N1(C(CCN(C2CCC2)CC#C)=O)CCOC(C(=O)NCC(=O)NCC)C1 CCCC(C)(O)CC(=O)N1CCCC(C)(CNC(C2CN(C)CC(C)O2)=O)C1 C(C(=O)NCC(C)NC(=O)CCc1cn[nH]c1)(C(C)C)NC(C)=O c1(C(=O)NC2C(NC(=O)C=Cc3ccco3)CCC2)nc2cnccc2s1 c1(OC)ccccc1-c1cn(CCCC(=O)N2CC(C)(C(N)=O)C2)nn1 CC(C)C(CO)CCNC(C1(NC(=O)Cc2ccccn2)CCN(C)C1)=O C1(N(C(C(C=C)O)=O)C)CCN(C(c2ccc(Br)cc2)=O)CC1 c1(C(N2CC(C)(C)C(C(=O)NCCn3cccn3)C2)=O)cccn2ccnc12 N1(C(C(C)=C(CC)C)=O)CCC2CCN(C(C3CC4CCC3CC4)=O)CC2C1 C(CC(C)(C)NCC1(CCN)CC1)(c1nnnn1Cc1ccco1)OCC c1(C(N2CCC(C(=O)OC)C2)=O)ncc(F)c(=NCc2ccc(O)c(C)c2)[nH]1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NC1CC1CNC(=O)CC1CCCO1 Cc1ccnc2sc(C(=O)N(C)CC3(CNC(=O)C4=COCC4)CC3)c(C)c12 N1(C(c2n[nH]c(C)c2C)=O)C2CCCC1CC(NC(=O)C=CC(C)C)C2 CCC(C)C(C(=O)NCC(C1CC(C)(C)C1)O)N(C)C(c1n[nH]c2c1COC2)=O c1(SC)c(C(=O)NC2CCOC(c3cccs3)C2)cccc1Cl c1(C(N2CC(O)(CNC(C(CCOC)C)=O)C2)=O)cc(OC)cc(C(F)(F)F)c1 Cc1ccn2nc(C(N3CCC(C4(NC(c5cc(C)sn5)=O)CC4)C3)=O)nc2n1 C1(CC)(CC)CC(C(=O)NC(C)CC2CN(C(c3c[nH]nc3Br)=O)C2)C1 C(=O)(C(CN(C)C)C(C)C)N1C(C(=O)NCc2cc(C)sc2C)(CC)CCC1 C(C(C)(O)C(=O)NCCCOCCC(=O)NCCc1ncnn1C)OC N1(C(C(C(C)C)F)=O)CC2CC1CC2CNC(=O)Cc1c(Cl)cnn1C c1(C(=O)NC(CNC(C(C)N(C(C)=O)C)=O)(C)C)ccc(F)c(CN(C)C)c1 CC(CC(=O)NC(C1CCCCCC1)CNC(c1nocc1C1CC1)=O)C(F)F C1(CNC(C=C(COC)C)=O)C(C)CCCN1C(c1cc(C)sn1)=O N#Cc1cc(F)c(F)cc1NC(C1CC(F)CN1C(c1sc(Br)cc1Br)=O)=O CC(C)CC(CNC(C1CC1C)=O)NC(=O)CN1CCS(=O)CC1 N#Cc1cccc(CC(=O)NCC2CC2NC(C2CCCCS2(=O)=O)=O)c1 N1(C(CC2C(C)=CC=CC2)=O)CC(C)CCC1.c1(S)cc(=N)[nH]cc1Br c1(C(=O)N)ccc(OCC)cc1.C1C(F)CNC(=O)CC2(CC2)C(=O)N1.CCOC.OC C1(C2CC2)(NC(c2csc(C)c2C)=O)CCN(C(=O)Cc2cccc(F)c2)C1 C1(COC)(CNC(=O)CCCC2CC2)CCCN1C(c1cc(Br)c[nH]1)=O n1(CCC(=O)NC2C(NC(C(C)NC(CC)(C)C)=O)C2)nc(C)cc1C c1(OC)cc2ccccc2cc1CN1CCC(O)C(C(=O)N(C)C)C1 c1(NC(=O)NCC(CC)C(F)(F)F)ccc2c(c1)CCCS2 c1(CNCC2N(C(CCc3c(C)ncs3)=O)CCOC2)cc2ccccc2[nH]1 c1(C(=O)NCCCN(C(C(CCC#C)O)=O)C)cccc2c1CCCN2 n1(CC)nc(C(N2CC=CC2CNC(c2c(OC)noc2C)=O)=O)cc1C c1(C(N2C(C(=O)Nc3c(C(C)=O)scc3)CCCC2)=O)ccc([Si](C)(C)C)cc1 C1(C(N(CC(=O)NCCC2CCC(C)O2)CC)=O)CC2(CSC2)C1 C(=O)(C(CNC(=O)CCC(C)(C)F)CCC)NCc1cccc(CC=C)c1 C12(C(=O)NCCCCN(C(C3N(CC)CCC3)=O)C)CCC(OC)C1CC2 C(=O)(CC(C)CC(C)C)NCC1(C)N(C(Cc2c(C)cc(O)cc2)=O)CCC1 c1(C(N2CCC(F)(C(=O)Nc3nccc(I)n3)C2)=O)cc(Cl)c2cn[nH]c2c1 c1(C(N(C2CN(C(C3(S(C)(=O)=O)CC3)=O)C2)C)=O)cnc(-c2ccncn2)nc1O CCCN=C(NCCc1cc(Cl)ccc1OC)NCC1C(CO)C1(F)F C1(CNC(CCCC=C)=O)CCN(C(=O)CCc2cccc(F)c2)C1(C)C C1(CNC(c2cc(C)nc(O)n2)=O)CC2(CCN(C(c3ccon3)=O)CC2)CO1 c1(N(C2CC3(CNC3)C2)C(Cc2c(C)cco2)=O)ncnc2c(Br)c[nH]c12 n1(CC(=O)Nc2cccc3sncc23)c(=O)cnc2ccccc12 C1(NC(CSCC(=O)N(CCN(C(C)C)CCO)C)=O)CC2C=CC1C2 N1(C(CCCOC(CC)=O)=O)CCN(C(c2cc(OCC)n(C)n2)=O)CC2(CC2)C1 C1(CNC(CSCCCC)=O)CN(C(=O)C(O)C2CC2)CC(C)(C)C1 c1(OC)ccc(CC(=O)NC2CN(Cc3ncc(CO)s3)CC2O)cn1 Cc1nn(C)c2c(NC(c3ccoc3)C)nc(N3CCc4[nH][nH]c(=N)c4C3)nc12 N1(C(=O)Cc2ccco2)CC(CO)C2(C1)CN(C(=O)C1=CC3(CCOC3)C1)C2 c1(C(=O)NC(Cc2ccc(F)nc2)C(=O)O)ccc(Nn2ccnc2)cc1 C1(CNC(=O)CCCF)CCN(C(c2ccc(CCO)cc2)=O)C12CCC2 C12(NC(C(C3CCN(CCC#C)CC3)C)=O)CCC(C1)OC2C c1(C(N(C2CN(C(=O)CCn3ccnc3)CC23CC3)C)=O)cc2ncccc2[nH]1 S(=O)(=O)(c1cc(C)cnc1N(C(CO)C1CC1)C)N(C)Cc1ccc(OC)cc1 N1(C(CC2CCC(=O)O2)=O)CCCCC1CCNC(C1CCC(F)(F)C1)=O C1(CC(=O)N(CC(C)CNC(C2(C(F)F)CCC2)=O)C)CCCCC1 O=C1Cc2c(N3CC4CCC(C3)N(Cc3cc(I)ccc3O)C4)ncnc2N1 CC(CC(=O)N1CCC(C)(NC(=O)C(O)C(F)(F)F)CC1)P(C)(C)=O C(c1ccc(Cl)cc1Cl)=C(c1nnnn1C1CCC1)NC(C1C2COCC12)C C=C1CC(C(F)(F)F)(C(=O)NCC2CCN2C(=O)CSc2cnn(C)c2)C1 CC1=C(C(=O)NC2(CN(C)C(c3nc(C)nn3C)=O)CC2)CCC(C)(C)C1 C1(CCNC(C(C)NC(CC)=O)=O)CCCCN1C(=O)CCc1ccc(C)s1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)Cc3nn(C)cc3Cl)c(=O)n2[nH]1 CC(C)(C#N)CCC(=O)NCC1CN(C(C2Cc3cccnc3C2)=O)C1 C1(CNC(C(C)(C)F)=O)(NC(=O)C(F)=CC2CC2)CCC(F)(F)CC1 CCC(C)(C)CC(=O)N1CCCC1C(=O)NCc1oc(COC)nc1C N1(C(CCC#C)=O)CCN(C(C2C=CC2C(=O)OC)=O)CC1CC(F)F c1(C(N2C(CCNC(Cc3c(C)nccc3)=O)COCC2)=O)ccc(=O)n(C)n1 C1(CC(=O)NC2CC(CC(=O)NCc3csnn3)C2)CCC2(CC1)CCC2O N1(C(c2ccon2)=O)CCN(C(=O)CCc2csc3ccccc23)C2CCCC12 C1(NC(c2cncc(C)n2)=O)C2COCC1CN(C(=O)C=CCOC(C)(C)C)C2 Cc1cnc(C(N2CCCOC(CNC(=O)Cc3cn[nH]c3)C2)=O)cc1Br N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CN(C(=O)C(N3CCOCC3)C)CC2C1 C1(C(CN(C)C(c2ccc(CC)cc2OC)=O)=O)CCc2nccn2C1 c1(COC)ccnc(C(=O)NCC23CC2CN(C(=O)C=CC2CCC2)C3)c1 C1(OC)CCCC(CNC(=O)C(C)(C)N(C(=O)CCC(C)C)C2CC2)C1 c1(-c2nc(Cc3nc(C)on3)n(C3CCCC3(C)C)n2)nccn2nccc12 c1(CC(=O)NCC(CNC(CC=C)=O)CO)ccc(S(N)(=O)=O)s1 c1(C(=O)NC2CCC(CNC(C(C)=C(CC)C)=O)C2)cc(OC)cc2c1OCC2 C(=O)(CC(F)(F)CCCC)NC(CNC(C(CC=C)C)=O)C1CCC1 c1(C(N2CC(C)C(NC(=O)C3=CCCOC3)CC2)=O)ccc(C#N)cc1O N1(C(C2C(CC)C2)=O)CCC(C(=O)N(C)Cc2nc(C)ns2)C1C c1(C(N2CCC(C)(CNC(CC(CC)C3CCC3)=O)C2)=O)cnc(OC)c(C)n1 N1(C(c2c(C(C)=O)ccnc2)=O)CCCCC(CNC(c2cc(C(N)=O)co2)=O)C1 N1(C(CC2(C)OCCO2)=O)CCCC(C)(NC(=O)C(F)CC2CCOC2)C1 c1(C(N2C(Cc3cn(C(CC)C)nn3)COCC2)=O)cc(S(N)(=O)=O)ccc1Br N1(C(c2ccc(CC)cn2)=O)C2CCC1C(NC(=O)Cn1cc(C)cn1)C2 c1(N(C)C)cccc(Br)c1CN1CCNCC1C(=O)NC(C)(C)CO c1(C(=O)NCCCN(C(=O)C(c2cccnc2)O)C)cc(=O)c(Br)c[nH]1 C(C)(CCC(=O)N(CCCCCNC(c1ccnc(S)c1)=O)C)OC C12(NC(CC3CCCC(OC)C3)=O)CCCC1N(C(C1(C)CC=CCC1)=O)CC2 C1(CNC(CCNS(CC)(=O)=O)=O)CCN(C(=O)CN(C2CCC2)C)C1(C)C CC1(C(=O)NCC2CC3CCC2N3)OCCc2ccccc21 N1(C(CCS(C)=O)=O)CC2CCC1CN2C(c1ccc([N+](=O)[O-])s1)=O C(CSC)(C(=O)NCC1OCCC1C(=O)NC1COCC1N(C)C)OC N1(C(C2(C=C)CC2)=O)CCC(C2CCN(C(=O)C(C)SC(F)(F)F)CC2)C1 c1(C(=O)NCC2(C(=O)Nc3cncc(Br)n3)CC2)cccc2c(Br)n[nH]c12 C1(CC=C)(NC(c2csc(S)n2)=O)CCN(C(C2CCCC23CC3)=O)C1 CC1CCC(NC(c2ccc(F)o2)=O)CN1C(C1CC(c2ccccc2)C1)=O N1(C(c2nn(CC)c(O)c2)=O)CC2CC(NC(c3n[nH]c(C)c3O)=O)C2C1 c1(C2(C(=O)NC3CN(C(C(C)OCC=C)=O)C3)CCOCC2)cccc(C#N)c1 c1(CNC(=O)CC2OCCCO2)cccc(NC(c2ccc(F)o2)=O)c1 C1(C(=O)NCC2(OC)CC(C)C2)CC12CCN(C(=O)CC1CCSC1)CC2 CC1(C)COCCC1NCCNC(=O)CC(C(F)F)n1cccn1 c1(C(N(CCC(C)NC(COC(C)C)=O)C)=O)cnc2c(c1)c(O)nc(=O)n2C Cc1ccc(C(=O)NC2CC(C(=O)Nc3ccc(Cl)c(Cl)c3Cl)C2)c(I)c1C C1(CNC(C2CC2c2cccc(C(F)(F)F)c2)=O)CCCCC1c1cccc(F)c1 Cc1cc(F)cc(NNC(=O)COCC2(C(F)(F)F)CC2)c1 C(=O)(C1CCc2cc(F)ccc21)NCC(C)N(C(COCCC=C)=O)C c1(C(=O)NC2CCCN(C(c3nnc(CC)s3)=O)CC2)c(O)nnc(C)c1C C1(COC)CC2C1CCN2c1nnc(-c2ccc(Cl)nc2)n1Cc1ccccc1 S(=O)(=O)(c1ccc(Cl)cc1)N1C(C(=O)NCC(CC)(CC)OC)CCC1 Cc1cc2c(C(=O)NCCC3CN(C(=O)CCc4cnn(C)c4)C3)nccn2n1 CCC(CC(=O)NCCC1(O)CCN(C(c2c(Cl)csc2Cl)=O)CC1)C(F)F C#Cc1ccc(C(N2CCCC2C2(NC(=O)C(O)C=C)CC2)=O)cc1Cl N1(Cc2cncc(OC)c2)CC2(CCN(C(=O)C(C)(C)F)CC2)C1 C(=O)(C(CO)NC(N)=O)NCCOCCN(C(=O)C(C)(C)c1ccno1)C N(C1c2ccccc2CC12CCCC2)c1cc(N2CC(CCF)OCC2)ncn1 c1(CC(=O)N(C2CCN(C(=O)C(F)(F)c3cccnc3)C2)C)ccc(F)cn1 C1(NC(CC2(C#N)CC2)=O)C=CC(C(=O)NCC2COC(=O)N2)C1 C1(NC(CCCNC(C)=O)=O)COC2C(NC(c3nc(C)c(C)s3)=O)COC12 N1(C(c2c(C(=O)OC)scc2)=O)CCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C(F)C1 Cc1nonc1NCC(F)(F)F.C1(C)(CNC(=O)CC(=O)N(C)C)CCC(=O)N1 Cc1c(C(=O)NCC(O)CN(C(=O)Cc2cccc(C(N)=O)c2)C)cccc1F c1(C(N2CC(SC)C(NC(C3OCC4CCC34)=O)C2)=O)c(O)cc(Cl)cc1F N1(C(C2C(NC(C(C)C(F)(F)F)=O)COC2)=O)CC2C3CCC(C3)C2C1 n1(CC(N2CC3C(CNC(C4C(CC)C4)=O)(C3)C2)=O)ncc(C#N)c1N N1(C(Cc2c(C#N)cccc2)=O)CC2(CCC(C(N3CCCC(F)(F)C3)=O)O2)C1 c1(OC)cccc(C(C)=CC(=O)NCCN(C(=O)CC23CC(C2)C3)C)c1 C(=O)(CCCCCC(C)O)N(CCNC(C1(OC)CC(C)CC(C)C1)=O)C1CC1 CC1CN(C(=O)CC2COCCO2)CC1(C)CNC(=O)C=Cc1ccsc1 c1(CNC(C2CCc3n[nH]cc3C2)=O)cnn2cc(Br)ccc12 c1(CCN(C)Cc2cccc(Br)c2)ccc(CO)c(F)c1 C=CC1(CC(=O)N(C(C)CC(C)CC)C)CN(C(=O)C(C)NC=O)C1 CN1CCC(CCC(=O)NCC(C)(CO)NC(c2ccc(F)s2)=O)C1 c1(CC)cc(CC)[nH]c(=NCC2CCCCN2C(c2ccc(Cl)c(Cl)c2F)=O)n1 C1(C(N2CC(C(C)NC(=O)Cn3cccn3)C2)=O)CCCC1C1CC1 C(=O)(CCCC(F)(F)F)NC1(CF)CCN(C(C(C)C=Cc2ccccc2)=O)C1 CC1CCC=C1C(=O)NC(C1CN(C(c2ccc(Cl)c(Br)c2)=O)C1)C C(CC(C(=O)Nc1ccccn1)N1CCC(c2cccs2)CC1)N1C(=O)CCC1 c1(C(=O)OC)ccc(C=CC(N2CC(NC(C34CC(C)(CO3)C4)=O)C(O)C2)=O)o1 C1(n2cc(C(C)OC)nn2)CN(C(C2CC=CC(C(=O)O)C2)=O)CCO1 c1(C(C)(C)NC(C2CCOCC2)C(=O)OCC)n[nH]c(CCCl)n1 c1(C(=O)Nc2cnc(F)cc2C(=O)NCC(O)CO)ccc(O)c([N+](=O)[O-])c1 Cc1coc(C)c1C=CC(=O)NCCC1(C)CCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NCC2N(C(C#CC(C)C)=O)CC(C)CC2)ccc2cnoc2c1 Cc1cc(CNC(C2CCC(CNC(c3ccc(CO)o3)=O)C2)=O)sn1 c1(C(N2CC(C)(NC(C(n3ncc(C)c3)C)=O)C2)=O)ccc(C(=O)O)nc1O O=S(=O)(c1ccnc(C2OCCO2)c1)N1CCC(OC2CC2)CC1 C#CC1(NC(C2CC2CNC(=O)C=CCN(C)CC)=O)CC2CCCC12 C#Cc1cncc(C(=O)NCCCC(N2CC(S(C)=O)C2)=O)c1 C12(CC(=O)NCCNC(=O)C(C)Oc3ccccc3C(F)F)COC(CF)(C1)C2 c1(NC(CC2N(C(C=Cc3ccc(C)s3)=O)CCOC2)=O)cc(F)ccc1O N1(C(c2cc(C)cc(Cl)n2)=O)CCC2(CC1)CCN(C(C1COC(=O)C1)=O)C2 c1(NC(=O)NCC(O)CNC(C2CC2c2cccs2)=O)ncn2c1CCC2 C1(C(=O)NCC(c2c(OCCCOC)cccc2)(C)C)Cc2c(C)cccc2O1 C(C(C)(C(=O)NCCc1nc(C)no1)NC(=O)CCCn1cncn1)SC Cc1cc(F)ncc1C(N1CCC(CNC(=O)CCn2ccc(=N)[nH]2)C1)=O N1(C(C(COC)OC)=O)CCC2CCN(C(c3cnc(OC)c(C)c3)=O)CC12 N1(C(C(N2CCSCC2)C)=O)CCN(C(=O)CCCc2cncs2)C(C2CC2)C1 S(=O)(=O)(CCCN=c1[nH]c2c(c(=NCC3(OCCOC)CCC3)[nH]1)SCC2)NCC c1(C(N2CC3C(NC(C(C)SCCCC)=O)(C3)C2)=O)cnn2c1CC(F)(F)C2 c1(C(=O)NC2C3(NC(C(C)OC)=O)CCC(C2)C3)nc2ccccc2cc1Cl N1(C(=O)NCC(CC#C)C2CC2)CCC2(CC1)CC2CSc1cc(C)ccc1Br N1(C(c2[nH]ccc(=N)n2)=O)CC=C(CNC(c2ccnc(O)c2)=O)CC1 C1(CNC(CSC)=O)CN(C(c2c[nH]c(=N)s2)=O)CCC1(F)F C1(C(=O)NC2(CN(C)C)CCC2)CCCC(NC(=O)CC23CCCC2C3)C1 c1(C(c2n(C)nnn2)NC2CC2(C)C)cn(C)c(=O)c2cnccc12 CC1CCc2nc(S(=O)(=O)NCC(C)(C)OCCOCCO)cnc2C1 c1(CNC(c2cc3c[nH]cnc-3n2)=O)cccc2c1CCN(c1ncns1)C2 C(C(C)CC(=O)NOC1CCOC1)NC(c1c(CC)nn(C)c1)=O C1(CNC(CCCC(=C)C)=O)CN(C(=O)Cc2ccn(CC)n2)CCC12CCC2 N1(C(CCCN(C(=O)CC2CCCC(=O)C2)C)=O)CCC2(CC1)N=N2 c1(C(N(CCCN(C(C(C)OCCC=C)=O)C)C)=O)cc(C(C)(F)F)ccn1 C1(C(=O)NC2CC(OC)C2)CC2OCC1CN(C(=O)CN(C)CCOC)C2 C1(NC(C(N2CCOCC2)C)=O)CC(CNC(=O)CSc2ccc(Cl)s2)C(O)C1 C1(C(N2CCC(NC(COCC(C)(C)C)=O)C(O)C2)=O)CCC2(CCC2)CC1 C1(CCC)(NC(=O)CC2(N(C(=O)CCc3cccnc3)C)CC2)CCNC1=O CC1(C)CCC2(CCN2C(C2(O)CC2)=O)CC1 CC(CSc1ccccc1)C(=O)NC1CC(C)(CNC(=O)C(C)(F)F)C1 C12(C(=O)NCCOCCCNC(c3n[nH]c4c3CCC4)=O)OCCCC1C2(F)F C1(C(=O)NCC2CCN2C(=O)Cc2nc[nH]n2)CCOC1C1CC1 C1(C(=O)NC(C(=O)NCC)C(C)C)CCC2CCC1N2C(c1ccn(C)n1)=O c1(C2N(C(C3(c4cn(C5COCC5O)nn4)CCC3)=O)CC2)ccc(Br)cc1 CC1(C)CCCC(NC(C23CC2CN(C(C2(C(N)=O)CC2)=O)C3)=O)CC1 c1(C(N(C)CC2C3CN(C(C(C)C4CC4)=O)CC32)=O)ccc(Cl)c(F)c1 c1(C(=O)NCC(C)N(C)C(c2ccc(F)c(Cl)c2)=O)ccc(N)c2ccncc12 N1(C(C(C(C)C)SCC)=O)CCCC2(C1)CN(C(=O)Cc1ccn(C)n1)CCO2 c1(CC(C)NC(=O)SC(C(=O)NCCNC(c2ccoc2)=O)C)cncnc1 CCC(CC)(CC)C(=O)N1CC2CC1C2NC(C1OCC1(C)C)=O CCC(CC(=O)NCC1(N)CCCCC1)SC.C12(CCC1)C(=O)NC2.C(C)(C)OCO N1(C(CCc2n(C)c(S)nn2)=O)CCC2(NC(c3csc(C(F)F)n3)=O)CC2C1 N1(C(C2CC(=C)C2)=O)CC(C(=O)Nc2cnc(OCC)nc2)C(C)C1 c1(C(N2CC(CNC(C(C)(Cl)Cl)=O)OCC2)=O)cc(S(=O)(=O)NC2CC2)c[nH]1 C(CF)(C(=O)Oc1ccccc1)NCCC1(C(=O)NC2CC2)CC1.CN(C)C c1(CC(N2C(CNC(CCCSC)=O)C(C)CCC2)=O)c[nH]c2cc(Cl)ccc12 C1(NC(CC(CC)c2ccccc2)=O)CCC2CC1CN2C(=O)C(C)C1CCC1 N1(C(C(C2CCOC2)OC)=O)CCCC2(NC(c3nncn3C3CC3)=O)CC2C1 C1(C(N2CCC(NC(c3ccc(Cl)nn3)=O)C2)=O)C2C3CC4C1C1C2CC3C41 C1(C(C)NC(c2cscc2C(F)F)=O)CN(C(=O)CC2(N3CCCC3)CC2)CCO1 c1(C(N2CCC(C(C)NC(Cc3ccc(SC)cc3)=O)C2)=O)cn2ccnc2s1 c1(C(=O)NC2CC(O)C2)cccc2c1CN(Cc1ccn3ccnc3c1)CC2 c1(C(N(CC(C)N(C(C(CCC)C)=O)C)C)=O)ccc2cc(C)ccc2n1 c1(C(N2C(C)(CNC(=O)CCN3CCCC3)CCC2)=O)ccc(F)c(Br)c1F NC1CCOCC1CC(=O)NCC(F)(F)CN(C)C c1(C(=O)NCCCNCC2CC2)csc(NC(c2scnc2C2CC2)=O)n1.C C(=O)(C(C)CC(F)F)N1C(C(C)C)CCC1C(=O)NCC1(C#N)CC1 Cc1ccc(C(=O)NC(C2CCCN(C(c3cc(O)cc(F)c3)=O)C2)C)c(F)c1 C1(CC(c2nnnn2Cc2ncoc2C2CC2)NCCCSC)CC2C=CC1C2 N1(C(Cn2c(C)cc(C(=O)OC)n2)=O)CCN(C(=O)C2=CCOCC2)CC1C c1(OC)cccc(C2=NOC(CSC(=O)N=c3ccn(-c4cccnc4)[nH]3)C2)c1 O=CN1CCCC1C(=O)OCC12CC(C(F)(F)F)(CO1)C2.c12ccc(nn1)[nH]2 N1(C(CCNC(=O)C2CC2)=O)CC2(C(=O)Nc3cccc4nncn34)CCC1CC2 N1(C(=O)CC2CCCCO2)CCC2CCN(C(c3nccc4occc34)=O)C2C1 N1(CC)CCOCC1CC(N1CC(F)(CNC(c2cccc(N(C)C)c2)=O)C1)=O N1(C(CCCCC=C)=O)CC(C(N2CCOC(C(C)(C)C)C2)=O)C2(CCC2)C1 C12(N(C(c3nc(Br)cs3)C(=O)NCCSC)C)CC(C)(C1)OC2(C)C C1(C)(CC)CC(NC(c2c(F)cccc2F)=O)CN1C(c1cncnc1C)=O C(=O)(C(O)C(F)(F)F)N(CCNC(c1n[nH]cc1CC1CCCO1)=O)CC1CC1 C(CCCC(=O)NCC1CCCC1C(=O)NC1CC(O)C1O)SC C[Si](C)(C)C1(C(N2CCCC2C2CCCCC2O)=O)COC1 c1(C(C(C)NC(=O)NCCCCc2ccccn2)OC)ccccc1F c1(C(N(C2CCN(C(C3CC3(F)F)=O)C2)CC)=O)cc2nc(=O)ccn2[nH]1 N1(C(C=C(C)c2ccccc2)=O)CCC2(CC2)CC1C(=O)Nn1ccnn1 c1(NCc2ccc(N(C)C)nc2)cnc(F)cc1C(=O)NCc1cscn1 N1(C(c2cccc(SC)c2)=O)CCC(NC(=O)C(=O)NCC2CC2)C12CCC2 NC1C=CC(NCC2CCCC2OCc2ccccc2)C1 c1(C(N2CCN(C(N3CCC(C)CC3)=O)C(C)C2)=O)coc2cc(O)ccc12 C1(CC(=O)NCC(=C)CC)CC(C)(C)CN1C(=O)CC(C)(C)O CON(CCC(=O)NOC(C1CCOC1)C1CC1)C(=O)C(C)CC(F)(F)F c1(C(=O)OCC)ccc(C#N)c(Cl)c1.C1CC2CCC1(NC(=O)C(F)CC1CC1)C2 N1(C(c2c(C)nsc2N)=O)CCC=C(CNC(=O)Cc2ncn(C)c2C)C1 N1(C(COCCCCC)=O)CCCC1C1(NC(=O)CN(C)C(=O)OC)CC1 N1(C(CC2(C)CCCC2)=O)CCC(O)(CNC(c2cc(C3CCC3)[nH]n2)=O)C1 N(C1CC(C)n2ncnc21)C(c1n(C(C)C)ncc1)c1nnnn1C(C)(C)C CC(C)CCCCC(=O)N(C1CCC2CN(C(C3(C)CCSCC3)=O)CC12)C N1(N(CC(Cl)Cl)C)CC=C(C(=O)NC)CC1.C1(C=O)CCC(C)(C)C1 C1(C(=O)NC2C(C)=C2)CCCC(NC(=O)CCCOC(C)(C)C)C1 N1(C(C2CC(C)(C)C2)=O)CCC(CC(N)=O)(NC(c2cn[nH]c2)=O)CC1 C(C)(CO)(C(=O)NCC(C)(C)CNC(=O)CSC(F)(F)F)OC C(C(CC1CC1)C(=O)Nc1cnccc1SC)NC(C(C1CCC1)OC)=O C(N=c1[nH]c(NC2CC(=O)NC(=O)C2)nc2c1CCC2)C1C(c2cn(C)nc2)C1 N1(C(c2cc(OC)c(Cl)cc2)=O)CCC(C)C(NC(c2cccnc2)=O)C1C C(=O)(CC(C)CC(C)(C)C)NCC(CC=C)C(=O)N1CCN(CC)CC1 c1(C(N2C(C(=O)NC(CC=C)CO)CC3CC32)=O)c[nH]c2nccc-2c1 c1(C(=O)NCC(CNC(c2ccn(C(C)C3CC3)n2)=O)(C)O)cnc(Cl)n1C C1(NC(c2n(CC)c(O)nc2)=O)CCN(C(=O)CCC2CCCOC2)CC1(C)C c1(C(N(C(C)CCNC(C2CCC(C)O2)=O)C)=O)cccn(C2CCC2)c1=O CC1C(NC(=O)Cc2ccccc2)CCN1C(=O)COC1(C)CCC(C)C1 N1(C(C2N(CC)CCC2)=O)CCCC(CC)C1C(=O)NC(C)CCSC c1(-c2cn(C)c(=O)cc2)nc(C(=O)Nc2cccc(C#N)c2Cl)n2ccccc12 N1(C(C=Cc2n(C)ncc2)=O)CCN(C(=O)CCc2cncs2)C(CO)C1 N1(C(CC2C(C)=NNC2=O)=O)CC2(C(=O)NCCN3CCCC3=O)CC1CCO2 CCC(CCCO)N=c1[nH]c(N2CCOCC2)nc(=NCc2cnn[nH]2)[nH]1 C1(NC(C=CC)=O)CC=C(C(=O)NCC(C)(C)OCCO)C1 N1(c2c(C(N3CC4=C(CCC(C)(C)C4)C3)=O)cccc2)CCC(O)C(F)(F)CC1 C(=O)(C1=NOC(C)C1C)NC1C(SC)CN(C(=O)CC2CCCO2)C1 c1(NC(c2ccccc2F)CNC(C(C(C)C)NC(C)=O)=O)ncccc1C#N n1(CC(=O)NCC(CNC(CC2C(CC)C2)=O)OC)cc(Cl)c(C)n1 c1(CN2CCCC(CNC(=O)CN(CCO)CCO)C2)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)NC2CN(C(C(c3ccc(C)cc3)=O)=O)C(C)C2)cc(O)nc(O)n1 C(CC(C(=O)NCC1CCCO1)NC(=O)CCOCC(C)(C)C)=CC C(C(O)CC(F)(F)F)N(CCNC(c1ccccc1N1CCOCC1)=O)CC Cc1cccc2c1CCN2C(c1occc1CNC(c1coc(C2CC2)n1)=O)=O C#CCC(C(=O)NC1CC(=O)N(C2CC2)C1)NC(c1csnc1Cl)=O N#Cc1ccc(O)c(NC(=O)C(C2CCOC2)NC(c2cc[nH]c2)=O)c1 c1(OC)ccc2[nH]cc(C(=O)NC3CCOCC3NC(C3CSC3)=O)c2c1 C1(C)(CC)CCC(CNC(=O)C(C)(CO)NC(c2csnc2OC)=O)O1 c1(C(N(CCOC)CCNC(c2cc(C)sc2C)=O)=O)cncn(C)c1=O N=c1nc(Cl)cc(C(N2CCCC(CNC(C3CCCN3C=O)=O)CC2)=O)[nH]1 Cc1nn(C)c2cncc(C(=O)NCC34CNC(C)(C3)C4)c12 CCC(CC)CC(=O)NC(C)C(C)(C)NC(=O)CCC(C)(C)C Cc1c(NC(=O)C(=O)N(C)C(c2cccc(Cl)c2)C)cccc1Cl CC1CCC2(CC1)CCN2CC(=O)NCc1ccc(F)c(Cl)c1 C1(C2CCC2)(C(N(C)CC2(CNC(=O)CCCn3cncn3)CC2)=O)CC1 N1(C(C=CC(C)(C)SC)=O)CCCCC1C1CCN(C(c2ccc(Cl)s2)=O)C1 C1(OC)CN(C(c2ncc(F)cn2)=O)CC1NC(=O)CCc1ccc(Cl)nc1 c1(N(C2CCN(C(c3nc[nH]n3)=O)C2=O)C)cccc(N)c1F N1(C(C(C)CO)=O)CC2(COC(CNC(=O)COc3ccccc3F)C2)C1 Clc1cscc1CNC(c1ccnn1CCI)c1nnnn1-c1ccccc1 c1(-c2cn(C(c3ccccn3)CC)nn2)ccc(OCCNC)c(-c2ccccc2)c1 Cc1cc(C(N2CCCC(NC(C3CC3C(F)F)=O)C2)=O)c(C)n1CCO Cc1cc(=NC(=O)CN(C(C)(C)C)C(c2cccc(F)c2C)=O)[nH]o1 c1(CCC(=O)NC2CC3CN(C(=O)C(F)n4cccn4)CC23)c(F)cccc1F N1(C(c2cn(CC)nc2C)=O)CCC2(NC(=O)CCN(C)C(C)=O)CC2C1 C(=O)(C(C)(C)CC(F)F)NCC1C(NC(CCN(CCC)C)=O)CCCC1 c1(C(N(C2CCCN(C(C=CC(C)(C)C)=O)C2)CCO)=O)cccc([N+](=O)[O-])c1N C1(O)(CCNC(c2n(CCC)ccc2)=O)CCN(C(C2(SC)CC2)=O)C1 C1(CNC(C=CC(C)(C)C)=O)CN(C(=O)C(c2cccc(Cl)c2)O)CC12CCC2 CCS(=O)(=O)CC(=O)N1CCC(n2cc(-c3ccccc3O)nn2)C1 C#CCCCCC(=O)N1CC=CCC1C(=O)NCC1(C)CC2CCC1C2 C1(NC(C(c2ccoc2)NC(C(C)CO)=O)=O)CCCC(C2CC2)C1 c1(C(N2C(CNC(c3c(C)cnnc3)=O)C=CC2)=O)ccc(Br)c(F)c1 C1(NC(c2cncc(N)n2)=O)CN(C(=O)CCC2CC2(F)F)CC12CCC2 c1(NC(C2C3CN(C(C(CCC)CCC)=O)C2C3)=O)ccc2c(c1)OCCO2 c1(C(=O)NCC#CC(=O)NC(CO)C2CC2)c[nH]ccc1=O N#Cc1cc(C(c2nnnn2CC2CCCO2)NCC2OC3CCC2C3)cs1 C1(C(N(CC(=O)NCCC(O)CO)C2CCC2)=O)CCNC(=O)C1 c1(CN(C(CN2CCN(C)CC2)=O)Cc2c(I)ccnc2F)cc(Cl)cc(Cl)c1 C12CN(CC1F)CCn1nccc1C(=O)N2.c1(C)cc(Cl)sc1Cl.CO CCC(CC)CC(F)C(=O)NC(C)CC(=O)N(C)CC1CCCN(C)C1 c1(NC(C(C=C)OC)=O)ccc(C(N2CC(N(C)CC=C)C2)=O)cn1 c1(C(N(CC(C)NC(=O)CN2CCNC(=O)C2)CC)=O)cc([N+](=O)[O-])c(C)s1 C1(NC(C(CC=C)C)=O)CC12CCN(C(=O)CC1CC(C(C)=O)C1(C)C)C2 CC(CF)C(=O)NCC(C)(C1CC1)NC(=O)CSS(C)(=O)=O C1(NC(=O)Cc2cccs2)CN(C(=O)CCc2ccc(Br)cn2)CC2CC12 c1(OC)ccc(C(=O)NCCC2(O)CCN(c3ccncn3)CC2)cc1F C1(NC(C2CCN(C(CN(C)C)=O)C2)=O)(CO)CCCCC1 N1(CC23CCN(CC2)C3)CCC(CO)=C(F)C1.O=C1C2=NOC(C2)C(=O)N1 c1(C(=O)NC2CC3(CC(CNC(CCC#CC)=O)C3)C2)scc2c1OCCO2 C1(C(=O)OC(C(N2CCC(C)(c3ccccc3)C2)=O)=O)C2CCC3C(C2)CC13 C#CCC(C)(C)C(=O)NCC1(F)CCC(CNC(=O)C(C)(C)CCOC)C1 CS(=O)(=O)c1cnn(CCNC(=O)C(=O)NC2CC2(F)F)c1 c1(C(N2CCC(CC(C)(C)C)C2)C(=O)NCCCSCC)cc(Br)nn1CC CCC(CC)(O)C(=O)NCC(C1CC1)NC(c1sc(F)cc1C)=O CC1CCCC=C1C(=O)N1CCC2CN(C(c3ccc(F)cc3Cl)=O)C2C1 N1(C(C23C(NC(c4c(C)csn4)=O)C4CC2C3C4)=O)CCOC2(CCC2)CC1 N1(C(CC)=O)CCCCC1C(=O)NC(C1CN(C(C2CN(C)C2)=O)C1)C C1(C(N2CCC(CNC(C(COC)O)=O)C2(C)C)=O)Cc2ccc(F)cc2O1 C(=O)(C1=C(C#N)CCC1)NCC1CCCC(NC(c2ccc(C)s2)=O)C1 CC(C)(CCNC(c1cnccc1C#N)=O)C(=O)N1CCC2(CCC2)C1 C(=O)(CC(C)C(C)C)N1CC(OC)C(C(=O)N(CCO)CC2CC2)C1 C1(NC(C(N)=O)=O)COC2(CCN(C(c3cc4cccc(F)c4o3)=O)CC2)C1 C(C)(C)(CCCNC(=O)CC(c1c(C)noc1C)C)NC(CSCCC)=O Cc1nn(C)c(C(N2CC3CN(C(c4c[nH]cc4C)=O)C3C2)=O)c1Cl c1(CCC(=O)NCC(C(C)C)NC(C23CCCN2CCC3)=O)ccc(Cl)c(F)c1 c1(C(=O)NC(CNC(CCC(CC)OC)=O)COC)cc2nccnc2cc1F CC1(C)C2CCC(C2)C1NC(C1COCC1NC(=O)COc1ccccc1)=O C1(C(N2CC(C(C)(C)C#N)C2)=O)CCCCN1C(c1ccc(Cl)cc1)=O C1(C(=O)NCC2(C(N3CCCC(C)C3)=O)CCCO2)CC2C(C1)C2(F)F c1(NC(N2CC(CCC)C2)=O)ccn2nccc2n1 CC(C)C(F)(F)CC(=O)N1CCC1CNS(=O)(=O)C1CC1.N1CCC1C=O N1(c2cncc(OC)n2)CCCCC(CNC(=O)C=CCN(C)C)C1 C(C(=O)NCc1ccc(Cl)c(Cl)c1)(C(CC)CC(C)C)N(CC(=O)OC)CC#N c1(N(C)C)ncccc1C(=O)NCCCOCCC(N1CCC2CC2C1)=O C(=O)(C(C)(C)C(C)(C)C)NCC(CC(C)C)NC(c1cc(C)c(C)o1)=O C(=O)(C1COc2ccccc21)NC1CCCC(NC(C(CSC)(C)C)=O)C1 CCC(CC)(CCC(=O)NC1CC(C)N(C(c2nocc2Br)=O)C1)[N+](=O)[O-] C(=O)(C(CNC(=O)C(C1CC1)OC)CC1CCCC1)NCCN(CCCC)C C(c1ccccc1)=C(OC)C(=O)NCC(C)NC(=O)CCc1cncn1C C1(CNC(C(c2ccccc2)SCC)=O)CN(C(C2CCN2C)=O)CC1(F)CO c1(C(N2CC(CNC(CC(CC)O)=O)N(C)CC2)=O)ccc2c(C)[nH]nc2c1 C1(NC(C)=O)CCCN(C(=O)CCn2cc(-c3ccc(N(C)CC)nc3)nn2)C1 c1(NC(C2CNCCN2Cc2cc(Br)ncc2F)=O)ccnc(Cl)c1I N1(C(C2C(NC(Cc3cnc(C)s3)=O)CCC2)=O)CCOCC1C1CC1 Cc1oc(C(=O)NCC2(C)OCCCO2)cc1CO c1(C(=O)NC2(CO)CCN(C(C(C)OCC#C)=O)C2)cc(=O)c(Br)c[nH]1 c1(C(N2CCC(CNC(c3c(OC)scc3)=O)C2(C)C)=O)nc2ccccc2[nH]1 c1(N2CCC(C(C)(C)C)(CO)C2)nc2cccnc2c(=NC2CC2)[nH]1 N1(C(C2CC(C)N2C(C23CCC(C2)C3(C)C)=O)=O)CC(CO)C2(CC2)C1 C1(C(N2CCC(OC3CCN(C)C3)C2)=O)C2CC1N(C(C1(C)CC(C)(C)C1)=O)C2 N1(C(Cc2ccc(C)o2)=O)CCN(C(=O)CC2=CCCC2)C2CCCCC12 c1(C(=O)NCC(C2(O)CCN(C(CCN(C)CC)=O)C2)C)scc2c1OCCO2 C#CCCCCC(=O)NCC1C=CCN1C(c1ccccc1CO)=O C(=O)(C1=NOC(CNC(c2cnnc(O)c2)=O)C1)NCCC#CCC C(=O)(CCC(C)(C)C#N)NCC1(COC)CN(C(c2ccnc(OC)c2F)=O)C1 CC1CN(C(c2ccc(F)c(Cl)c2)=O)CCN1C(=O)CC1CC1C C=CC1(C(=O)NCCCCC(CO)NC(=O)CCn2ccnc2)CCOCC1 S(=O)(=O)(c1cnn2ccc(=NCCc3nc(=N)[nH][nH]3)[nH]c12)NCCCC(C)C c1(CC)conc1C(=O)NCC(CC)NC(=O)C(F)(F)C1CCOCC1 N1(C(=O)Cc2cccc(Br)c2F)CCC2CN(Cc3ccc(C4CC4)cc3F)CC12 C1(NC(c2nc(CC)oc2)=O)CN(C(c2c(Br)cncc2Br)=O)CC12CC2 CC(C)C(O)C(=O)N1CCC(C)(CNC(=O)CCc2cccc(O)n2)C1 C(=O)(N=c1cnc(Br)c(Cl)[nH]1)C1CCCC(NC(c2cccnn2)=O)C1 Cc1cc(Cl)ccc1OCC(=O)NCC(C)N(C)C(C1CCC(C)(C)C1)=O C(CCC)(CCC)=CC(=O)NC(CC=C)CNC(C1(OC)CCC1)=O Cc1c(C(=O)NCCOC2CCN(C(=O)CCS(N)(=O)=O)CC2)cccc1F C1(NC(=O)CC2C3CN(C(=O)CN4CCNC4=O)CC23)CCN2CCC1C2 N1(C(C2(CC)CCCO2)=O)CCC2(CCCN(C(=O)Cc3cc[nH]n3)C2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC2CC(O)C1C2NC(c1c(OC)csc1)=O c1(CCC=C)ccc(C(=O)NCC2C(CNC(c3occc3Cl)=O)C2(F)F)cc1 c1(C(N(C(C)C(=O)N(C2CC2C)C)C2CC2)=O)ccc(F)s1 N1(C(CC=CCC)=O)CCCC(C)(CNC(c2ccncc2C(=O)NC)=O)C1 N1(C(C2CC(=C)C2)=O)CCC(CN(C)C(c2cn(CCC)nn2)=O)C1 c1(C(=O)NCC(CNC(c2ccc(C(N)=O)o2)=O)O)cccc2ncnc(O)c12 N1(C(C2CCCN(CC)C2)=O)CCC2(CCCN2C(=O)C=Cc2csnc2C)C1 C12(C(=O)OCC)CCC(NC(c3cc(Cl)cnc3F)=O)(CC1)C2 c1(C(N(C2CC(NC(C(Cc3c(C)cccc3)C)=O)C2)C)=O)ccc(F)c(Cl)c1 C1(CCN(C(CCC=C(C)C)=O)C)CCN(C(C23CC(C2)C3)=O)CC1 O=S(=O)(c1cn[nH]c1)CN1CCCC1Cc1ccccc1F C1(NC(c2c(C)nc(O)s2)=O)CCN(C(c2cc(Cl)ccn2)=O)C1(C)C C1(C(N2CCC(F)C2)=O)(OC)CCCCC1.C1(=O)CC(C)(C)C2CN1CCN2 CN1CCC(CNC(c2cc(C3CC3)ns2)=O)C1c1ccc(F)cc1 C1(c2ccccc2Cl)(C(=O)NC2C(NC(C3(CCC=C)CC3)=O)C2)CCCCC1 C(c1nc2ccccc2s1)=CC(=O)NC1CCC1NC(C1CCC=CCC1)=O C1(C(=O)OC(C(C)C2C(CC(C)C)C2)=O)C2CCCCCC12 C#Cc1cnn(C)c1C(=O)NC(CC(C)C)C(=O)NCC12CCC(CO1)C2 c1(C(=O)OC)ccc(NC2CCNC2c2ccccc2)c(F)c1 c1(NC(C2C(NC(C34CC(C(=O)OCC)(C3)C4)=O)C2)=O)cn2cccc(C)c2n1 c1(NC(CC)(CNC(=O)CC2CC=CCN2C)CC)ncc2ccnc-2[nH]1 C1(NC(CCCN(C(C)C)C)=O)COCCN(C(C2CC2c2ccccc2)=O)C1 C(=O)(CC(=O)NCC1(C(=O)Oc2ccccn2)CCCO1)OC c1(OC)ccc(C(F)(F)F)cc1CC(=O)NC1(CC2CCCOC2)CC1 C12(C(=O)NCC3CCCN(C(C(CCC)(C)O)=O)C3)CCC(OC)(CC1)CC2=O CCC(C)CC(=O)N1CCCCC1CCNC(=O)Cn1cnc(C(N)=O)n1 CCCCC(=O)C(=O)N1CC(C(=O)NC(C)CC(CC)CC)CC(C)C1 Cc1cc(C(N2CCCC(N(C)C(C3C4COCC34)=O)C2)=O)nn1C C1(CN(c2nccc(NC)n2)CCCC2(CCOC)CCC2)CCC2(CCC2)O1 c1(CCC(=O)NCC2(C)CCN(C(=O)C(F)(F)C(F)F)C2)cc2ccccc2o1 CN1C(=O)CCCc2cc(C(=O)NC3(C4CC4)CCNCC3)ccc21 N1(C(CCc2cnn(C)n2)=O)CCCCCC(NC(c2n[nH]cc2Cl)=O)C1 c1(C(C)C)cnc(Cl)[nH]c1=NC1CN(C(=O)C(C)n2ccnc2)CC2(CCC2)C1 c1(CN2C(C(N3CCC(O)C(F)C3)=O)CC(F)C2)c(Br)cccc1[N+](=O)[O-] C1(CNC(C(C2CCCCC2)C)=O)CN(C(c2cnc(O)n2C)=O)CC1O C1(CNC(c2cncc(OC)n2)=O)CCN(C(c2nocc2C(C)C)=O)C(C)C1 C1(NC(C2C(C(=O)OC)C2)=O)CCN(CCOc2ccccc2)C1 c1(OC)ccc(Cl)cc1C(=O)NCC(C)(C)CN(C)C(C1CCOC1C)=O C(CC(=O)N(C(CO)C(C)C)C)(C(C)C)NC(C(C)NC(CC)=O)=O Cc1scc(C(=O)NCC(O)CN(C(=O)CN2CCN(CC(F)F)CC2)C)c1N C(CC(C)(C)C(=O)NCC(C)O)NC(c1c(C)cccn1)=O N1(C(C(C)OCC)=O)CCC(CNC(c2coc(Br)n2)=O)(OC)C1 c1(C(=O)NC2CCC(N(C(c3cc(C)sn3)=O)C)C2)c(Cl)ccc(C)c1N C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCC(CC)(CC)CO)(C)CSC c1(OCC(N2CC(O)(CN(C(CC=CC)=O)C)C2)=O)ccc(C)cc1C CS(=O)(=O)c1ccc(C(=O)OCc2ncccc2C(F)F)o1 CCN=c1cc(C(=O)NC2(CNC(=O)C(F)(F)c3csc(C)c3)CCC2)cc[nH]1 c1(SC(C)C(=O)OC(c2ccc(NC(C)=O)cc2)C)cc(=O)n2c(C)cccc2n1 C1(CCCC(=O)NC(C(=O)Nc2sc(CC)c(C)n2)CO)COCCC1(C)O C1(CCNC(C2C(C)(C)COCC2)=O)CCN(C(C2(O)COC2)=O)CCC1(F)F C(CCN=C(NCCC(C)(C)C)NC1C(C)(C)C1(C)C)SC N1(C(=O)CSC(F)F)CCOC2(CCN(C(C3CCCN3C3CCCC3)=O)C2)C1 O=C1c2ccsc2CCC1CC(=O)NCC1CN(C(=O)C=CC2CCC2)C1 c1(CC(N2CC(NC(C(C(C)C)NC(C)=O)=O)C2)=O)ccccc1S(N)(=O)=O N1(C(C(C(C)C)NC=O)=O)CC2OCC(NC(c3cccc(F)n3)=O)C2C1 Cc1ncnc(C)c1CC(=O)NCC1CC1CNC(=O)C(N1CCOCC1)C C1(CNC(C2C(C=C)C2)=O)CCCC12CCN(C(c1ccccc1F)=O)CC2 c1(C(N(CC(=O)Nc2ccc(Cl)c(Cl)c2)C)=O)cccc(S(C)(=O)=O)c1 N1(CC)CCCC(NC(C2COCCC2NC(c2cc(O)n(CC)n2)=O)=O)C1 c1(C(=O)NCC(C)NC(C2(CCC)CCNC2=O)=O)ccnc(O)c1F Cc1cc(C(=O)NCC(C)NC(=O)CC2NC(=O)NC2=O)n(-c2ccccn2)n1 C(=O)(CC1=NN(C)C(=O)C1)NC1C(CC)CN(C)C1.c12cccnc1NC2=O CC(C)C(CCCC(=O)O)NC(c1ccc(-n2cc(C(C)(C)O)nn2)cc1)=O CC1=C(C(=O)NC(C2CC2NC(C2CC(F)(F)C2)=O)C)CC1 C1(CNC(=O)CCc2cnco2)CC2(CCOCC2)CN1C(=O)CCCC1CC1 c1(C(N2C(C(=O)Nc3c(I)ccc(C)n3)CSCC2)=O)ccc([N+](=O)[O-])cc1C Cc1ccc(C(N2CCC(C)C(NC(=O)CCSC(F)(F)F)C2)=O)cc1C#N Nc1cccc2c1ccn2CC(=O)OCCCCC1CCCC1 n1(C(C)C)ccnc1-c1cn(C2CC(NC(=O)CC3C=CCC3)C2)nn1 c1(CCC(=O)NCCC2N(C(C3CN(C(=O)NC)C3)=O)CCC2)nnc(C)n1C c1(CNC(CC(CC)N(C(=O)CCC(C)(C)N(C)C)C)=O)ccc(F)c(O)c1 c1(CNC(C=CC(C)NC(=O)COC2(CO)CCCC2)=O)ccc(O)c(F)c1 c1(OC2C(OC)CC2O)cccc(CS(=O)CC2CC2)c1 N1(C(c2cnc(C)n2C)=O)CCC(NC(c2cnc(O)cc2O)=O)CC1C1CC1 C1(CNC(C2C(C(C)NC(=O)CC(C)N(C)C)C2)=O)CCCCC1O N1(C(CCNc2ccc(C)cc2)=O)CC2CN(C(c3ccc(I)c(C)c3)=O)CC12 Cc1nc2cc(C(=O)NCC(C)COC(C)C)cc(O)c2o1 Cc1nc2cc(C(=O)NC3CCCC3(C)CNC(=O)C=CCF)ccc2o1 CS(=O)CCC(=O)NCC1(CNC(=O)C=CC2CC2)CC1 CC1(NC(c2cc(F)ccc2F)=O)CCN(C(C2CCCCN2N=O)=O)CC1 C1(CNC(C2C=CCN(C(c3cnn(C)c3Cl)=O)C2)=O)CC2(CCC2)CO1 C1(CN(C)C(c2ccoc2C2CC2)=O)COCCN1C(=O)CCc1ccccn1 N1(C(c2c(CC(C)C)n(C)nc2)=O)CCC(NC(C2(C)CCC2)=O)C(CO)CC1 N1(C(c2cc(CC)no2)=O)CC2(C1)CN(C(c1cccc3scnc13)=O)CCO2 Cc1cc(C)c(C(N2CC(CNC(c3cnc(C)o3)=O)C3(CCC3)C2)=O)c(C)n1 N1(C(C(C)=C2CC2)=O)CC(CNC(=O)COCC2CCOCC2)CC12CCC2 C1(NC(C(CC)C)=O)CC12CCN(C(c1c(C)nc(=N)[nH]c1C)=O)CC2 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CO)NC(C(C(C)(F)F)(C)C)=O C1(CC(=O)NC2CCN(C(C3C(F)(F)C34CC4)=O)CC2F)CCC2(CC1)CC2 C(=O)(C(C)C(=O)OC(C)(C)C)NCC1(C(C)NC(CCC=C)=O)CC1 C1(O)(Cn2cc(CSC)nn2)CCN(C(=O)C(=O)CC2CCCO2)C1 CC1(C)CC=C(C(=O)NC2CC3CC2CC3C(N2CCC2CO)=O)CC1 Cc1ccc(CC(=O)NCCOCCNC(c2occc2C)=O)c(Br)c1 C(=O)(CCN=c1[nH]ccs1)NC1CCCN(C(C2C(C)C2)=O)CC1 C1(C(=O)NCC(C(=O)NC)O)CC(C)CN(C(=O)CC(C)(C)O)C1 c1(CC(=O)NCC2(NC(c3ccc(C(F)F)o3)=O)CCOC2)csc2nccn12 CCCCC(CC)CC(=O)N(CCC(N1CCCC2(CO)CCCC12)=O)CC C1(C(N2CCC(C)N(C(=O)Cc3cnn(C)c3)CC2)=O)CCC2(CC1)OCCO2 N1(C(CCC)=O)CCCN(C(=O)Cn2cc(Br)cn2)CC1.C1(O)CC(C(=O)C)C1 C1(NC(CCC(=O)NCCC)=O)CCN(C(=O)C(OC)OC)CCC1CO C=C(Cl)CC(C(=O)NCC(CN(C)C)CO)NC(=O)CNC(C1CC1C)=O C1(C)(CC)C=C(C(=O)NCCN2CCN(C(C3(Br)CC3(F)F)=O)CC2)C1 c1(C(=O)OCC)cc(O)nc(CNC(=O)NC2(C3CC3)CCOC2)n1 CC1(C)COC(C)(C(=O)NC2CCCN(C(=O)Cn3cnc(=N)[nH]3)C2)CO1 c1(C(=O)NC2(CF)CCN(C(c3nccnc3Cl)=O)C2)cc2c(s1)CCCC2 C1(CNC(CC(CC)C2CCC2)=O)CC2CCC(C1)N2C(=O)C(C)c1cccs1 c1(C(=O)NCC(C)CNC(=O)C(C)(Cl)Cl)cc2cc(O)ccc2[nH]1 N1(C(COCCCCOCC#C)=O)CCN(C)CC1CNC(=O)C(CO)OC(C)=O CCCC(CC)C(=O)NC1CCC(C)N(C(=O)CCn2ccnc2C)C1 c1(C(N2CCN(C3CCN(C(=O)C=CCO)CC3)CC2)=O)cccc2sccc12 C1(F)(CNC(C2C(c3cn(C)nc3)C2)=O)CCC(NC(=O)C(=O)NC2CC2)C1 c1(CC)c(C(=O)NCc2cncc(C(=O)NCCOC(C)CO)c2)ccn1C Cc1ccc(C)c(OC(=O)Nc2cnc(I)c(O)c2)c1 N1(C(Cc2ccc(OC)cc2)=O)CC2(CNC(=O)C=C3CCCC3)CCC1CC2 c1(C(=O)NC2(CNC(c3c(C)cco3)=O)CCCCC2C)ccc2nncn2c1 CCCCCC(O)CC(=O)N1CCCC1CCNC(c1ncsc1CC)=O Cc1nccc(Cl)c1C(N1CC(CCn2cc(-c3ccnn3C(C)C)nn2)C1)=O c1(CC)nc(CNC(N2CCC(c3noc(C)n3)CC2)=O)cc(O)n1 N1(C(CC2C(C)C2)=O)CCC(CCNC(c2csc(Cl)c2)=O)C1 c1(NC(c2scc(C(=O)Nc3c(I)ccc(C)c3)n2)=O)cc(F)cc([N+](=O)[O-])c1 N(C(=NCCC1=CCCCC1)NCc1ccco1)Cc1nc(C(=O)OCC)on1 CCC(CC(=O)N1CC(C(N2CC(C)(C)CC2C)=O)C(C)(C)C1)C(F)F C1(C(=O)NCC2C(C(=O)NCCc3c(C)ncs3)CCO2)CC12CCOCC2 c1(CNC(C23N(C(c4c(C)nc(CC)o4)=O)CCC2C3)=O)ccc(O)cc1C c1(C(=O)NC(C)CCNC(C2(CF)CCC2)=O)ccc(Br)nc1O C(=O)(C1=CCC(NC(c2sc(F)cc2C)=O)C1)NC(C#C)(C)C1CC1 c1(NS(CCCC)(=O)=O)c(C)cccc1F.C12CCN(C1)CC(=O)NC2C c1(C(=O)NCCNC(CCCC2CCC(C(N)=O)CC2)=O)cc(O)ccc1Cl c1(C(=O)OC)cccc(NC(c2cc(I)ccc2Br)=O)c1OC C1(CNC(C(C2CCC2)NC(CN(C)C(=O)C2CC2)=O)=O)CCC(C)(O)CC1 N1(C(C23N(C(C4CCN(CC)CC4)=O)CC(C2)C3)=O)CC2CCCCC2C1C c1(CCC(=O)NC(CN(C(C2C(C=C)CC2)=O)C)(C)C)ccnc(Cl)c1 N1(C(CCC=C(C)C)=O)CCCC(NC(=O)Cc2cc(C)no2)CC1 c1(C(=O)NC(C(C)NC(CC2(C=C)CCC2)=O)C)cc(C)c(C)c2ncccc12 Cc1c(NC(C2CCCN(C(=O)CN3C(=O)CNC3=O)C2)C)ncn1C.C(C)S N1(C(c2cn(CC)nc2C)=O)CC2(CC2)CC1C(=O)NC(C)(C)CC1CCC1 C1(C)(C(=O)NCCCN(C(C2CC2(C)C(F)(F)F)=O)CC)CC=CC1 N1(C(C(C)OC2CCCC2)=O)CCC(C2(NC(c3cc(Cl)c(Cl)[nH]3)=O)CC2)C1 N1(C(C(C(C)C)SC)=O)CCC(C)N(C(C2CC23CC(O)C3)=O)CC1 Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)NC1(C)CCCC(F)(F)C1 C1(CNC(=O)CCC2CCCO2)C2CC1N(C(c1ccc(C3CC3)nc1)=O)C2 C(CCC(O)C(=O)N1CC(S(C)=O)C1)NC(C1CC(C)N(C)C1)=O C12(NC(C(C)CO)=O)COC(CNC(C3CC(N4CCCC4)C3)=O)(C1)C2 c1(CC(=O)NC2CC(C(=O)NCC3CCC=CO3)C2)ncccc1F Cc1oc(C(=O)N(C2C3CN(C(=O)C(C)(C)CO)CC23)C)cc1CO c1(OCC(=O)NC2CC(NC(Cc3nnc(C)o3)=O)C2)ccc(C(C)(C)C)cc1 n1(CCOC)nnnc1C(C1CC1(C)C)NC(=O)CCSC(C)(C)C C1(CNC(=O)Cn2ncnn2)CN(C(=O)C2=COCC2)CC1C(F)(F)F O=C(CCCC1CCCO1)NCc1cc(C(=O)N(C2CCOC2=O)C2CC2)no1 C(=O)(C(CC(F)F)N(C(=O)C=Cc1cc[nH]c1)C)N(CCC(N)=O)CC C12(NC(C3CC(O)(CC#C)C3)=O)CCN(C(=O)CCC3CCCC3)CC1C2 C1(CNCCN(CC)CC)CN(C(=O)CCCCCO)CCC12CCC2.C(CO)O CC#CC1CCN(C(=O)C(C2CCC2)NC(C2COCC2(C)C)=O)CC1 c1(C(=O)NCCCOC2CCN(C(CC3(C)CC3)=O)CC2)cnc2[nH]ncc2c1 CCC(CC)(CN=c1[nH]nc(C)o1)NC(c1cn(CC(N)=O)nn1)=O Cc1ccc(C(=O)NC2CCCCN(C(c3ccn(CC#N)n3)=O)C2)cc1F c1(C(=O)NC(CN(C(c2cnc(OC)s2)=O)CC)C)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)NCC2CN(C(C3ON=C(C)C3)=O)CC23CC3)cc(F)c(C)cc1Cl N1(C(CNS(N)(=O)=O)=O)CCC(CNC(=O)C(F)CC2CCCC2)C1 c1(COC)nc(-c2cc(C3CC3)no2)n(C2COC(C)(C)C2)n1 C(CCCCC(=O)NC(c1nn(C)cc1O)C)NC(C1CC(C)SCC1)=O N1(C(CCCn2c(C)ncc2)=O)CCN(C(=O)C(C)C(C)(C)C)CC1CO C1(F)(CNC(C(CO)OC)=O)CCN(C(C2CC(F)(F)C2)=O)CC1 c1(CN(C(COC(C)C)=O)C)ccccc1S(N)(=O)=O c1(C(N2CC3(CCN(C(COCCCOC)=O)C3)C2)=O)cc2c([nH]1)CCC(C)C2 c1(C(=O)NCC2(OC)CN(C(CCN(C)CC)=O)C2)cc(OC)c2c(c1)OCO2 C(Cc1ccccc1)(C(O)C(F)F)N(C(Cc1c(OC)cccc1)=O)C N1(C(CC(c2ccccc2)SC)=O)CCN(C(=O)CC23CC(C2)C3)CCC1C C1(N(C(Cn2c(C)ccn2)=O)C)CCCN(C(C2(C)CC3CCC2O3)=O)CC1 CCC(C)(C)CCCC(=O)NCCC1(C)CCN(C(C2CCOC(=O)N2)=O)C1 c1(C(=O)NC(C2(CN(C(C)C)C)CC2)C)cc(OCc2ccccc2)cc(Br)c1 CCC(CC(=O)NC(CC(=O)NCc1ccon1)CC(C)C)C(C)(C)C O=C(C(O)CC(F)(F)F)NCCC1(O)CN(C(c2cc(Cl)cs2)=O)C1 CC(COC)CN1CCCC1.C(=O)(C(=O)NC1(C(=O)NC)CCC1)NCC(F)F C1(NC(c2cnc[nH]2)=O)CN(C(c2cnc(C3CC3)[nH]2)=O)CC1c1ccccc1 C1(C(=O)NCC2(NC(c3c(C(=O)OC)cco3)=O)CC2)CN2CCN1CC2C c1(C(C)NC(=O)CSCc2cncs2)ccc(F)c(F)c1 C1(F)(CNC(C=C(C)C(C)C)=O)CCN(C(c2cc(C(N)=O)cn2C)=O)CC1 N1(C(C=C(C)C)=O)CC(NC(C2(C(F)F)CCOCC2)=O)C(c2cnn(C)c2)C1 CC1CN(C(=O)Cn2nnc(=N)[nH]2)CC1(C)CNC(c1ccc(=O)n(C)n1)=O N1(C(C2CC2F)=O)CCOCC1CC1CC1.C12CN(CCO1)C2=O C1(CC)CC(C(=O)N(CC(C)C#N)C)C1.C12CC1CC(=O)NC2 N1(C(C=C(C)CNC(C2COC(=O)N2C)=O)=O)CCCC(C)(CO)C1 Cc1ncnc(C)c1C(=O)NC1CC(CNC(C2(CF)CC3(CCC3)C2)=O)C1 N1(C(CS(N)(=O)=O)=O)CC2CC1CCC2NC(c1cc2c([nH]1)CCC2)=O c1(CNC(C(CC)NC(=O)C(C2CC2)SC)=O)n[nH]c2c1CCC2 Cc1nc(CO)sc1C(=O)NC1CCC1NC(=O)C(O)Cc1cnn(C)c1 C1(C(=O)NCCC2(NC(c3c(OC(C)C)nccc3)=O)CC2)CC1C1(C)COC1 CC1CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)CCN1C(C12CCCC1C2(F)F)=O c1(OC)nn(C)cc1C(N1CCCC1CNC(=O)C(F)(F)c1ncccn1)=O C1(OCCNC(C=CC(=O)OC)=O)CCN(C(C2CC23CCC3)=O)CC1 C(Cc1ccccc1)(C(=O)NC1CCC1)OC(C)C#N C1(C(=O)NCC(CC(C)C)NC(c2c(C(C)=O)ccs2)=O)CC=C(C(C)C)CC1 C1(NC(=O)CC(Cl)Cl)CCN2CCC1C2.CC1(C)CNC(=O)CO1 c1(NC2CC(NC(C(CC)C(C)O)=O)C2(C)C)cc2nnc(C)n2cn1 C(=O)(CC(C)C(=O)NCC1CCC(C)CN1C(c1ccc(C)n1C)=O)OC N1(C(C(CC)=O)=O)CC(F)CC1C(=O)Nc1ncc(Br)nn1 CCC(C)C(C(=O)NC1CC2(C1)CC(C(=O)NCc1cncc(C)c1)C2)N(C)C N1(C(C2N(CC)CCC2)=O)CC(CNC(c2cncnc2C(C)C)=O)CC1(C)C N1(C(CCCNC(C)=O)=O)CC2(C1)CN(C(C1CC(Cl)(Cl)C1)=O)C2 n1(CC)cnc2[nH]c(=NC3CCC=CCC3)[nH]c(=NC3CCOCC3OC)c12 c1(CC)ccc(C(=O)NC(C)(C)CCCNC(=O)C(N2CCNC2=O)C)c(Cl)c1 CC(N=c1cc[nH]cc1)C(=O)N1CCCC12CCN(C(=O)CC(C)(C)O)C2 C1(CC(=O)OC)(C(=O)NC2CCC(NC(=O)C=CC3CCCO3)C2)CCCC1 Cc1nnc(Cn2cc(CNC(c3n[nH]c(CO)n3)=O)nn2)o1.C1(=O)CN1.C(N)(=O)N c1(OC)ccc2c(c1)CCN(c1nnc(NC(=O)CC(C)SC3CCCC3)s1)C2 c1(C(C(=O)N(CCN(C(C(C2CCOC2)OC)=O)C)C)(C)O)ccc(Cl)cc1 N1(C(c2c(C)scn2)=O)CCC(C2CCN(C(c3cc4cn[nH]c4cn3)=O)C2)C1 C1(NC(C2CCN(C(C)=O)CC2)=O)COC2(C1)CN(C(C1(C)CCC1)=O)C2 C(=O)(C(CN(C)C)C(C)C)NC(CC1CN(C(CCC(=O)OC)=O)C1)C C1(C(C)C)CN(C(=O)C(=O)NCc2cc(Br)ccc2Br)CC(c2ccccc2)O1 c1(CC)cc(C(N2CCCCC(NC(C3(CSC)CC3)=O)C2)=O)c(C)nn1 c1(C(=O)NC(CNC(C(CC)(C)OC)=O)(C)C2CC2)ccc(Br)cc1F C(=O)(C(C)(C)CS(C)(=O)=O)NCCCNC(C(C)N(C(C)=O)C)=O Cc1cccc(NC(C2(F)CCN(Cc3cc(C(=O)O)ccc3F)C2)=O)c1Cl C1(C(=O)NC2CCCN(C(C(C=CC)O)=O)C2C)CCOCC12CCCCC2 c1(C(CNC(CCSC)=O)NC(=O)C(C)OCCc2ccccc2)ccccc1 Fc1ccc2cccnc2c1-c1cccc(F)c1 c1(C(N(C(C)CNC(=O)C(C)(C)c2cscn2)C)=O)nccc2c1CNC2=O Cc1cc(C2(C(=O)N(C)CC3CCCN(C(C4CC4(Cl)Cl)=O)C3)CC2)cc(C)c1 c1(OC)ncc(C(N2CC3CC(Nc4cc(C)nc(C)n4)C3C2)=O)cc1Br c1(OC)ccc(CNC(C23CC2CN(C(N2CCC(C)CC2)=O)C3)=O)cn1 CC(C)CCC(F)C(=O)NCC(C)(O)CNC(=O)CNC(=O)C1CC1 CCC(C)(C)C(O)C(=O)N1CC(CCNC(=O)Cc2ccccc2)C1 N1(C(c2n[nH]c(C)c2F)=O)CCC(CNC(=O)CN2CCC(C)C2)C12CCC2 C(CC)(CCCO)N.C1(=O)CCCN(C(C)C)C(=O)CN1CCOC C1(=O)CCC2(CC2)N1.C(=O)(C=CC(=O)OCC)C=O.C1(CC)CCC1.C1CO1 C#Cc1ccc(C(N2CCOC(C3CC3)C2)C(=O)NC2COC2)cc1 C1(O)(C(=O)NCC(=O)Nc2ccccc2)CCN(C(C2CC2C(F)(F)F)=O)CC1 C(C1CN(C(C2(C)CC3C=CC2C3)=O)CC1C(=O)NC1CC(=C2CC2)C1)=CC C1(NC(C=C(CC)C)=O)CCC(NC(=O)C(c2cncc(F)c2)(C)C)CC1 CCCC(C(=O)N1CCC(C(=O)NCCc2cc(C)on2)(CC)C1)NC(N)=O C#CCC(C)(CC)C(=O)NCC1(CC(=O)NC(c2cnn(C)c2C)C)CC1 C1(NC(C2(C(C)C)COC2)=O)CCCN(C(C2CC(O)CN2C)=O)C1 C1(NC(C(C)OCCC(C)C)=O)CC(NC(c2c[nH]nc2C2CC2)=O)CC1O C1(C(=O)NC(C2CN(C(c3ccc(N)c(Cl)c3)=O)CCO2)C)CN2CCN1CC2 c1(NCCN(C(c2c(OC)ccnc2)=O)C)ncnc2sc(C)nc12 c1(C(=O)NCC(CNC(C(C)C2CCC2)=O)F)nc[nH]c2ncc(Br)c1-2 C(C(N=c1[nH]ccn2nnnc12)C(C)C)NC(c1nc(CCC)sc1)=O N1(C(C)C(=O)NCC(O)CNC(C2(CCF)CC2)=O)CCOCC1 c1(C(C(=O)NC2CCCOC2)N(CCC#N)C)coc(Br)n1 c1(-c2c(F)cc(OC)c(C)c2)n[nH]c2cc(C(N3CCCC3C(C)C)=O)ccc12 Cc1cc(=O)n(CCC(=O)NCC2CC(O)CN2C(=O)C(C)CC(F)F)cn1 C1(NC(C2(CC#C)CCN(C(c3cc(=O)cc[nH]3)=O)C2)=O)CCC2CC1C2(C)C c1(C(C)=O)ccc(C(N2CC(CCNC(=O)C(C)(C)c3cnsc3)C2)=O)cc1 C1(CN2CCC(NC(C(N3C(CC)CC3)=O)=O)CC2)CCCCCCC1 N1(C(C(C)OCCc2ccccc2)=O)CCC2(CN(Cc3ccncc3Cl)C2)C1 N1(C(c2c(CC)noc2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 N1(C(c2cc(C)oc2C)=O)CC2CCOC2(CNC(C2CCN(C)S2(=O)=O)=O)C1 C1(C(C)(C)O)CC2CN(C(=O)C(O)C3CC3)CC12.C1(=O)CO1 C(=O)(C(CC)CC)NC.c12ccccc1CC(=O)NCCOC1CCN(C1)C2=O CC1CN(C(c2cnc(S)nc2)=O)CC(C)N(C(c2ccc(Cl)c(F)c2N)=O)C1 N1(C(CNC(CC)(C)C)=O)CCOCC1CCNC(=O)C=Cc1ccccc1.CCOC c1(NC(c2ccc(CCC(=O)Nc3cccnc3Cl)[nH]2)=O)cc(Cl)ncc1Br CC(CC(=O)NC1CC12CC(NC(c1cncc(C(C)(F)F)c1)=O)C2)C(F)F C1(NC(c2c(C)ccn2C)=O)COC2C(NC(C34CCC(CO3)C4)=O)COC12 Cc1ccc(F)c(O)c1C(N1CCC(O)(C(C)NC(=O)C(C)CC(N)=O)CC1)=O N1(CCNC(=O)C=Cc2nccs2)CCCN(C(C2CCC2CF)=O)CC1 c1(CNC2C(C(=O)NCc3c(CC)ccs3)CCC2)ccnc(F)c1Cl c1(C(=O)NCC2CCN(C(c3n[nH]cc3Cl)=O)C2)cn2cccc(Br)c2n1 Cc1cnc2n1CCN(C(C)(Cc1ccccc1F)N(C)C)CC2 C1(C(=O)NC23CC(CNC(c4n(CCC)ccc4)=O)(C2)C3)CCC(C)(F)CC1 CC1(C)CC(CNC(C2CC(O)C2)=O)CN(C(=O)CC(C)(O)c2ccccc2)C1 c1(NCC(c2ccc(OC)cc2)OC)cc(P(C)(C)=O)ncn1 N1(C(CC2N(C(C)C)CCC2)=O)CCCC(C(N2CCCCC2)=O)C1 C1(CN(C(=O)CC2CCCCC2O)C)COCCN1C(C1C2CCC1CC2)=O C(=O)(C1=NNC(=O)C1)NCCN(CCC)Cc1nc(C)c(C)s1 C1(NC(c2ccc(C)nc2)=O)CN(C(=O)C=C2CCC(C)C2)CCC1CO Fc1ccc(-c2noc(C34CCCCC3C4)n2)c(OC2CC2)c1 c1(C(=O)NC2CN(Cc3ncccc3Br)CC2F)cc2n(n1)CCCC2 N1(C(C2CCC(C)(C)CC2)=O)CCC2CCC(NC(=O)Cn3cccc3)C12 CC(CCN=c1nc(CO)cc[nH]1)NC(=O)C(C1(O)CCOCC1)(F)F c1(OCC(=O)N(CCNC(=O)CC2CC3CC3C2)CC)cccc(F)c1 c1(CNC(c2ncc(OC)nc2)=O)ccc2c(c1)OCO2.C12CC(C1)CC(=O)N2 C1(C(C)NC(CC(C)O)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC1 C(=O)(CC(C)C(F)(F)F)NC1CC(CC(=O)NC(COC)(C)C)C1(C)C C=CCC(C)(CC)C(=O)NC1CCCC(N(C)C(c2cnc(OC)c(C)c2)=O)C1 N1(CC(=O)NC(=O)OC(C)(C)C)CCc2cc(-c3cncc(C(=O)O)c3)ccc21 c1(OCC)ncccc1CC(=O)NCC1(F)CC(NC(=O)CC2CCCO2)C1 C1(CCC=C)(C(N2CC(OC(C)C)C2)=O)CN(C(=O)C(OC)OCC)C1 N1(C(CCSCCCC)=O)CC(C(=O)NC(=O)C(CCC)N(C)C)CC1(C)C N1(C(CC2N(CC)CCC2)=O)CCC2CC1CN2C(=O)CCCN(C)C(C)=O S(=O)(=O)(c1csc(C2CCCO2)n1)N(CC(CC)O)Cc1ccccc1 c1(C(=O)NC2C(OC)CCC2)c(C)ncnc1C.C123CC(C1)(C2)NC3=O N1(C(c2n(CC=C)ccc2)=O)CC(CCNC(=O)C=C2CCSCC2)OC(C)C1 N1(C(C(CC#CC)NC(C23CSCC2C3)=O)=O)CC2(CCC(=O)N2)C1 c1(CN2C(C(=O)Nc3n(CC)ncc3)CCC2)ccc(OC)c(OC)c1 c1(C(=O)NC2CC3CC2CN3C(c2sccc2C2CC2)=O)csc2c1CCCC2 C1(NC(C2(NC(c3cc(Cl)cn3C)=O)C(C)C2)=O)CCCN2CCCC12 C1(OC)CCCCC1C(=O)NC(C)CNC(C)=O CN1CCCC1(C)C(N1CC(CNC(c2ncnn2C2CCOCC2)=O)C1)=O C1(C(=O)NC(C2(O)CN(C(=O)CCC3CCCC(=O)N3)C2)C)CC(F)C(=O)N1 C=CC(C(F)(F)F)NC(C1C(NC(=O)CCOCCN(C)C)C1(C)C)=O c1(N2C(CNC(C3C(SCC)CCC3)=O)CC(F)(F)C2)ncc(C#N)cc1Br C1(CNC(C(COCC)(C)C)=O)CC2CC(C1)N(C(c1c[nH]cc(Cl)c1=O)=O)C2 C(=O)(C(C)CC(C)CC(C)C)N1CCC(CCOC)(NC(c2cc[nH]n2)=O)CC1 n1(CCCC)nnnc1C(CC)(C1CC1)NC1(C2CCOC2)CC1 C12(CNC(c3c(C(C)(C)C)cccn3)=O)CCC1CCN2C(=O)CCC1CC1 CC12COC(C(=O)NCC(C)(C)NC(c3cc(C4CC4)[nH]n3)=O)(C1)C2 C12(C(=O)NCC3CCCN(C(c4n(CC)ccc4)=O)CC3)CCCC(CCC1)C2 N1(C(c2c(C)nc(CC)s2)=O)C(C)CC2CN(C(C3OCC4CCCC34)=O)CC12 Cn1c(O)nc2cccc(C(N3CC(CCNC(C4CCCC(O)C4)=O)C3)=O)c12 C(=O)(C1CCN(C)c2ccccc21)NCCC1C(C)CN(C(c2ccsn2)=O)C1 N1(C(C2CC(C)(C)C2)=O)CCC(F)(C(=O)Nc2oncc2C#N)C1 CC1(C(N2CCCC(CNC(=O)Cc3ccc(F)cc3)CC2)=O)CCNC(=O)C1 Cc1cc(N)ccc1C(=O)NCC12CCC1CCN2C(=O)CCCNC(N)=O C1(NC(c2ccc(C)s2)=O)CC12CCN(c1ncc3c(n1)CCC3)CC2 C(=O)(C#CC1CCCCC1)N(CC(CO)(CO)NC(=O)C=CC1CCOC1)C C(=O)(C(F)CCC(C)C)NC1CN(C(C=Cc2occ(C)n2)=O)CC(O)C1 N1(C(CCC#C)=O)CCCCC1CCC(=O)NCC(C)(C)C(=O)NC CCCCC(O)C(C)C(=O)N(CC(C)(C)CNC(=O)C(O)CCC)CC N1(CC(=O)NC2CC(C(=O)NCc3c(C(C)C)nn[nH]3)C2)CCNC(=O)C1 c12ccc(cc1)o2.c1(CC(=O)OC2CC(C)(OC)C2)ccc(O)nc1 C1(OC)CC(NC(c2ccc(C(F)F)o2)=O)CN(C(C2CC2Br)=O)C1 c1(N2CC(C)(C)C(NC(C3CC4CC4C3)=O)C2)c(Cl)cncc1[N+](=O)[O-] n1(C(C)(C)C)cnnc1C1CC1.c12cc([nH]n1)CN2.C1C(O)CCC(=O)N1 n1(CCC)cc(C(=O)NCCC2(CNC(C3CCCC3O)=O)CC2)nn1 N1(C(c2n(CC=C)ccc2)=O)CCN(C(c2cscc2C)=O)C(C)C1 Cc1nc(CNC2CC(C(N3CCC(CO)C3)=O)C2)co1 C(CC1=CCN(C(C2CC2F)=O)CC1)NC(=O)CCc1ccccc1Cl Cc1nc(Cl)ccc1C(N1CCCC(n2cc(CN3CCOCC3)nn2)CC1)=O C1(C2CN(C(C3CN(C(=O)NC)C3)=O)C2)(NC(C2(C(C)C)CNC(=O)C2)=O)CC1 c1(CC(Cc2cn(COC)nc2)C(N)=O)c[nH]c2cc(F)ccc12 c1(C(N2CCC(O)(CNC(=O)CCC3CCOC3)C2)=O)cnc2ncccc2c1 C(=O)(C(CO)C(C)(C)C)NCc1c(CCNC(C(C(C)C)NC(C)=O)=O)ocn1 N1(C(Cc2cn(CC)nc2)=O)CC(N(C)C(C2COC3(CCC3)C2)=O)C2(CC2)C1 C1(CNC(C=CCC)=O)(OCCNc2nnsc2C)CCOCC1 c1(C(N(CC(C)(C)NC(C2C(CC)OCC2)=O)C)=O)nc(C)n(C)c1C N1(C(CC)=O)CCC2(C1)CN(C(=O)C(C)NCS(=O)(=O)Cc1ccccc1)C2 N1(CC(=O)NCC2(NC(C3CC3F)=O)CC(OC)C2)CCNC(=O)C1 c1(C(C(=O)NCC(Cn2cc(CCNC(C)=O)nn2)(F)F)C2CC2)ccc(Cl)cc1 c1(Cc2n(C)ncc2)cn(C)nc1OCc1ccccc1.c1(C2CN2)ccccc1 C12(N(CCNC(COCC)=O)C(c3ccccc3CC(C)C)=O)CCCC1C2(F)F C(c1ccc(C)s1)=CC(=O)NC1C(CNC(C2(CC#C)CCCO2)=O)COC1 CC(F)CC(=O)N1CCC(CCNC(=O)CCCF)C1 c1(OC)ccc(S(=O)(=O)NC2CC(NCc3cnc(O)c(Cl)c3)C2)cc1OC C(=O)(C(O)C(CCC)NC(c1cc(C(F)F)[nH]n1)=O)N1CCC(F)(CCC)C1 c1(C)ccc(CC)cc1.N1(CC=C)CC2C(C(=O)NCc3cc(C)no3)C2C1 Cc1nc([N+](=O)[O-])cn1CC(N1CCN(C(=O)C(C)C)C2CC12)=O C#Cc1ccc(C(N2CCC(CC=C)(NC(=O)NC3CC3)CC2)=O)cc1 C1(N(C(=O)C(O)C2CC2)C)CC2CCC(C1)N2C(C1(C(F)(F)F)CCCCC1)=O N1(C(C2C(C(C)C)CCO2)=O)CC2CC1C2CNC(C1(N(C)C)CC1)=O C(=O)(C1c2ccccc2OCC1(C)C)N1C(C)CC(NC(=O)CC(C)(F)F)C1 C1(C(N2C(CNC(=O)CCNC(c3ccco3)=O)CC2)=O)(CF)CC(F)(F)C1 C12(C(N)=O)CCCC1(C(=O)NC13COC(CNC(C4(F)CCOC4)=O)(C1)C3)C2 CC1(C)CCC(C(=O)NC23CCC(C2)C3)(NCCOCCO)C1 c1(C(=O)NCC2C(NC(CN(CC)CC)=O)C2)cc(C)nn1C1CCOCC1 C1(CC)CCC(C)N(C(c2cn(C)c(=O)n2C)=O)C1.C12CN(C1)C2=O Cc1cccn(CC(=O)NCC2CC(C)CCN2C(C2C3COCC23)=O)c1=O CC1CN(C(=O)NCCc2cnco2)CC(C)(C(F)F)O1 C1(CN(C(=O)CC2C(NC(C3CCS(=O)CC3)=O)CC2O)C)CCC(C)(C)C1 C(=O)(CCCC(CC)CC)NCC(CC(=O)NC(CC#C)CC(F)F)OC c1(OC)ccc(C(C)C)c(C(=O)N(C)CCN(C(=O)C2=C(Cl)CCC2)C)c1 c1(C(=O)NC2CC(N(C(COCCCOC)=O)C)C2)cc2c(C)c(Cl)ccc2[nH]1 Cc1ccc2oc(NCC3CN(C(=O)CCN(C)CCO)CC3C)nc2c1 N1(C(c2c(C)cc(C3CC3)cc2)=O)CC2CCC1CC2NC(C1CC1(C)C)=O c1(C(=O)NCC(CC)NC(=O)CCC=C(C)C)cnc(C)[nH]c1=N C1(C)(CC)CCC(C(=O)NC2C=CC(CNC(C3(CC(C)C)COC3)=O)C2)O1 C1(C(N2CCC(NC(c3ccc(=O)oc3)=O)(CF)C2)=O)Cc2cc(F)ccc2O1 CCCC(C(=O)NCC(O)CC(=O)N(CCCCO)CC)OCC C1(C(=O)NCC(C)(C)NC(=O)CCn2cccn2)CC2(C1)CC2F C1(CC(=O)NCC2N(C(CSc3n[nH]c(=N)s3)=O)CCC2)CCCC(CCO)C1 C1(OC)CC(OC)CN(C(C2(C)CCCN2C(=O)CN2CC(=O)NC2=O)=O)C1 c1(OC)ccc(OC)c(C(=O)N(C)Cc2cn(-c3cc(C)cnc3F)nn2)c1 c1(NC(C)=O)ccc(CC(=O)NC(C)CNC(c2c(C)ncn2C)=O)cc1 N1(C(C(c2ccc(Cl)cc2)CC)=O)CCC(NC(=O)CN(C)C2CC2)C(C)(C)C1 N1(C(CC(C)c2ccco2)=O)CCN(C(C2CCC=CCC2)=O)CC(O)C1 c1(C(=O)NC(C)(C)C2CCC2)c[nH]nc1CCNC(=O)CCc1ccsc1 C1(NC(CCn2c(C)nc(C)n2)=O)CC2CC(C1)N(C(c1c(O)noc1C)=O)C2 c1(C(C)NC(Cn2ccc(C(C)=O)n2)=O)nn(C)c(=O)o1.C1C(=O)OC1 C1(CC)CN(C(C23CC(CCO2)C3)=O)CCN1C(=O)C(n1nc(C)cc1C)C C=CCC(CNC(=O)CNc1ccccn1)NC(=O)C(C)(C)C.C1(=O)CN1 CCCCC(F)C(=O)N1CCC(C=CC(=O)NC2(C)CCCC2O)CC1 C1(C(C)C)CN(C(=O)CC2CCCC(NC(C3CCC4(CC4)C3)=O)C2)CCN1C N#Cc1cccc(F)c1CC(=O)NCC1CCC1CNC(=O)CC1CC=CC1 C1(CN(C(c2cc(C(N)=O)[nH]n2)=O)CC)CCCCN1C(=O)C(C)CSC c1(C(=O)NC(C2CN(C(C3CCCC(F)(F)C3)=O)C2)C)ccc2c(O)n[nH]c2c1 N1(C(Cc2c(C)non2)=O)CCCC(NC(c2cscn2)=O)C1C c1(CN2CC(CNC(c3ncn(C)c3)=O)C2)ccc2ncccc2c1 C123COCC1CN(C2)C(=O)C(F)ONC3=O.C1(OC)CCC(CN(C)C)CC1 CC1(NC(=O)CCN2CCC2)CC(NC(=O)CCNC(c2ccco2)=O)C1 c1(C(N2C3C(NC(CC(C=C)CC)=O)C(C3)C2)=O)cc(C)cc2c1NCCC2C N1(c2nc(COC)nc(C)c2)CC2(C)CN(C(c3coc(COC)n3)=O)CC2(C)C1 c1(CC)nn(C)c(Cl)c1C(=O)NC1CCN(C(C2CC3CC2C3)=O)C1 c1(C(C)C)cccc(CC(N2CCN(C(=O)COCCN(C)C)CC2)=O)c1 C1(CNC(CCc2cc(C)no2)=O)CC(C)CN(C(C2(CCO)CC2)=O)C1 S(=O)(=O)(c1ccc(NC(C)=O)cc1)NCC1C(OC)C1 Cc1cc(C(=O)NC(CNC(=O)C(C)(C)c2cncs2)C(C)C)co1 Cc1cc(C2CC2C(=O)N(CCC(C)NC(c2cn[nH]c2)=O)C)on1 c1(CC(=O)NCCNC2N(C(=O)OCC)CC(O)C2O)c(C)nc2cccnn12 C=C1CCC(C(=O)NCc2nocc2C(=O)NC(C)(CO)CCF)CC1 N1(C(Cc2ncc(CC)[nH]2)=O)CCCC(C)C1CNC(C1(O)COC1)=O N1(C(Cc2ccc(OCC)cc2)=O)CCCC(NC(=O)C(F)C2CCOC2)C1C C12(CNC(c3ccncc3)=O)CC1CN(C(=O)CNC(C1CCCCC1)=O)C2 C(CCC(C)C(=O)N1CCCC(NC(c2nonc2N)=O)C1)OC C1(COC)(NC(C2CCCCC2C)=O)CCN(C(=O)C(C)(C)O)CC1 c1(C(N2CCC(C)(CNC(CC3(C)CCC3)=O)C2)=O)ccc2c(=O)ccoc2c1 c1(OC)noc(-c2nc(C3CCCC3)nn2-c2cn[nH]c2)c1Br C1(CNC(C2CSCO2)=O)CC2CCC1N2C(c1cc(Cn2cccn2)on1)=O C1(C(=O)NC2CC(NC(=O)CCCn3cccn3)C2)(OC)CCOC1 c1(C(N2CCC(N(C(=O)CCc3nc(C)no3)CC)C2)=O)cccc2nonc12 N1(C(c2c(C)cncn2)=O)CCCC1(C(=O)NC1(CO)CC2CCCC12)C(C)C N1(C(C2CCN(C(C3OCC(C)C3)=O)C(C)(C)C2)=O)CCCC12CCNC2=O C1(CC(N2CC(C)C(NC(c3cnn(C4CCC4)c3)=O)C2)=O)CCCCC1(F)F c1(C(N(C2CCN(C(c3cnn(C(C)(C)C)c3Cl)=O)C2)CC)=O)[nH]c(C)nc1C N1(Cc2c(C)nc(-c3ccc(OC)cc3)s2)C(=O)CCN(CC23CCCC2C3)C1=O c1(C(=O)NC(Cn2cccn2)C(=O)O)ccc(C(F)(F)F)c(Cl)c1 C1(C(N2CC(CN(CC(C)C)CC)C2)=O)C2CC(O)C(C2)N1C(=O)CSC c1(C(N(C(CNC(C2C(C)OC(C)C2)=O)C)C)=O)cc(O)cc(C#N)c1 c1(C(N2C(CNC(C3CC(OCC)C3)=O)CC3CC32)=O)ccc2cncn2c1 C(=O)(CC(C(F)F)n1cccn1)NCC(=C1CN(C(C2(C(F)F)CC(=C)C2)=O)C1)F C1(C(=O)NC2(C)CCN(C(Cc3c(C)scc3)=O)C2)CCCC2(CC2)C1 C1(CNC(CCCSC)=O)CN(C(=O)CCNc2ncccn2)C2CC12 C1(NC(CNC(c2cccc(C)c2)=O)=O)CN(C(c2cscc2F)=O)CC1(F)F c1(C(=O)NCCC=C)n[nH]c2ccc(-c3cnn(CCCNC(C)=O)c3)cc12 C(=O)(CC(O)CC(C)(C)C)N1CCCCC(N(C(C(=O)NCC)=O)C)C1 N1(C(CN(C)C)=O)CCC2CCN(C(c3cccn4[nH]c(=N)nc34)=O)C2C1 c1(C(N(CCOC)CCNC(C2CC(=O)N(O)C2)=O)=O)cc(CC(C)C)nc(O)c1 c1(CC(=O)N(CC(C(N2CCCC(COCC)C2)=O)O)C)ccc(C#N)cc1 c1(CNC(c2ccc(C)nc2)=O)nc2c(s1)CN(C(c1cscc1C#N)=O)CC2 C#CCC(C)(C)C(=O)NCC(CC=C)C(=O)N1CCC(n2cncn2)C1 CC1Cc2n[nH]cc2CN(C(=O)C(=O)N(C)CCc2ccc3c(c2)OCO3)C1 c1(C(N2CC3C(C(N4CCC(C)(C)CC4)=O)(C3)C2)=O)ccc2ccccc2n1 N1(C(Cc2ccc(C)nc2)=O)CCCC2CN(C(=O)C#CC3CCOCC3)CC12 C1(CNC(=O)COC(F)(F)F)CCN(C(C2(CO)CCCC2)=O)C12CCC2 CC(C)CC(C(=O)NC1CNC(=O)C1)NC(c1cccc(=O)o1)=O c1(OCC)ccc(C(=O)Nc2nccc(C#N)c2OC)c2ccccc12 c1(C(=O)NCC(CN(C(C(CC)(F)F)=O)C)O)cccc(F)c1C CN1CCC(c2ncc(C(=O)NCCOC3CN(C(=O)C=CC(N)=O)C3)[nH]2)CC1 C(=O)(CCC(=O)NC(CO)C(=O)NC(C1CCCC1O)C)NCCC Cc1cc(C(=O)N(CC(C)C(=O)NC(C)CC(N)=O)C)cnn1 N1(C(C2(C)CCC(F)(F)C2)=O)CC2(CCCN(C(c3nocc3Cl)=O)C2)C1 C1(NC(C(C)Cc2ccccc2Cl)=O)CC12CCN(C(C1CC(O)C1)=O)CC2 C1(NC(COCCCC#C)=O)CCN(C(=O)Cn2ccnn2)C2CC12 C1(C(C(=O)N(C2CN(C(c3ccc(OCC)cc3)=O)C2)C)C)CCC(C)(O)CC1 C(=O)(C1=C(C)CCC1)NCCCC(C)(C)NC(c1c(COC)cccc1)=O C1(=O)C2=NOC(C2)CN(C(=O)C(F)(F)CC=C)CCCN1.C(C)(C)(C)OCC c1(C(=O)NC2(C)CC(NC(c3cc4ccccc4[nH]3)=O)C2)cc(F)c(Cl)cc1Cl C1(S(C)(=O)=O)(C(=O)NCCN(C(=O)CC2CCCS2(=O)=O)C)CCC1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC(C)(CC(C)C)NC(=O)C=CS(C)=O CC(C)C(C(=O)NC12CC1CN(C(=O)CCCCn1ccnn1)C2)C1CCC1 C1(C(=O)NCC2(CNC(CC)=O)CCCC2)CCCCC1C1CC1 CC1CN(C(C23CC(F)(C2)C3)=O)CC(CCNC(c2cc(Cl)cn2C)=O)O1 CC1(C)CC(NC(=O)CCC2CCC(=O)N2)CN(C(C2(CS(C)(=O)=O)COC2)=O)C1 Cc1cnc(C(=O)NCc2ccc(C(=O)NC(C3CCOCC3)C)s2)cn1 N1(C(CCC=C)=O)CC(C(F)(F)F)OCC1CNC(=O)Cc1cccc(O)c1 C1(OC)CN(C(C2C(CCC)CN(C(C3CC4(CCC4=O)C3)=O)C2)=O)CC1(F)F C(=O)(C1CCC(=O)c2cccn21)NC1(CNC(C(C)OC2CCCC2)=O)CCC1 N1(C(COCCC#C)=O)CC2(C1)CN(C(C1CC1F)=O)C2 C(=O)(C1CCCc2cncn21)NC1CCC(NC(=O)CCc2cncs2)CC1 N1(C(=O)CC2COCCN2C(c2cccnc2Br)=O)CCc2ccsc2C1 N1(C(N(c2cnn(C)c2)CC)=O)CC(C)OC(C)C1C C1(CCN(C(C2N(CC)CC2)=O)C)CCCCN1C(=O)CN1CCC(F)CC1 N1(C(C(C)OC)=O)CCCC(N(CCO)C(c2ccco2)=O)C1.C1(=O)CN1 N1(C(c2snc(C)c2N)=O)CC(F)(F)CC1C(N1CCC1C1CCC1)=O c1(C(N(C2CCN(C(c3c(C)scc3)=O)C2)C)=O)ccnnc1N.C(C)C c1(NC(C2CC3CC3N2C(c2sc(Br)cc2Br)=O)=O)cc(Cl)cc(Cl)c1F c1(CC(=O)NCC2N(C(c3cccc(OCC)c3)=O)CC2)ccc(C)c(F)c1 CCC1(C)CC(=O)N1.C1(C(=O)OC(C)(C)C)CC(=O)N(C)C1c1cccs1 CC(N=c1ccnc(NCC(=O)Nc2cccc(Cl)c2Cl)[nH]1)C1CCCCC1O N1(C(=O)Nc2cnn(-c3cccc(C)c3)n2)CCCc2c(N(C)C)cccc21 C1(NC(c2ccnn2CC(F)F)=O)CCN(C(=O)C2=COCCC2)C12CCCC2 c1(C(=O)NCC(CO)NC(c2cc(-c3ccncc3)no2)=O)cccc(O)c1F C1(CNC(c2cnn3c2CCCC3)=O)CC2(CCN(C(=O)CCCCF)CC2)C1 C(=O)(CC(C(F)(F)F)N(C)C1CC1)NC(C)CCNC(c1cc(Cl)cc(F)c1N)=O C1(OC)CCC2CN(C(=O)CCCCNC(C3(C)CCC(=O)N3)=O)CC12 c1(C(=O)NC(CNC(c2ncn(C(C)C)n2)=O)C)ccccc1F c1(C(=O)OC)ccc(NC(=O)Nc2ccccc2N(C)C(C)C)cc1.C(C)(C)(C)O C1(C(N2CC(N3CC(F)C3)C2)=O)(NC(CCCOC(C)=O)=O)CCCC1C c1(C(=O)NC2C(CO)CCN(C(CCCOC(C)C)=O)C2)cc(Cl)c(Cl)cc1N Cc1c(C(=O)N(C)CC2CN(C(=O)CC3(C(F)F)CC3)CCO2)ccn1CCO C(=O)(C(O)CC[S+](C)C)N(C)CC1CCN(C(C2(CCC=C)CC2)=O)CC1 C(=O)(CC(C)C(F)(F)F)N1CC(NC(C(CCC#C)O)=O)C1 C1(NC(N2CCC(C)(c3n(C)ncc3)C2)=O)CC(c2nnco2)C12CCC2 C1(CNC(C(C2CCCC2)OCC)=O)(CO)CCCN(C(=O)Cn2cnnc2)C1 C1(C(C)NC(C(C)OCCOC)=O)CN(C(C2(C)CNC(=O)C2)=O)CCO1 c1(CC)cc(C(c2nnnn2C2(C)CC2)NCC2(C)CCCS2)ncc1F N#Cc1ccc(OCc2ncccc2NC(C2CCC(=O)C2)=O)cc1 C1(CCNC(Cn2cc(C(N)=O)nn2)=O)CSCCN1C(=O)CC1CCC=CO1 CCC(C)(CC)C(=O)NCC12CC(C1)C(NC(=O)CC1CCCC(C)(C)C1)CO2 C=CCC(CC)C(=O)NCCOCCN(C(=O)Cc1cc(C)cc(C)c1)C C1(Cc2cn(-c3nccc(C)n3)nc2)CC(=O)N(c2ccc(Cl)cc2)C1=O c1(SC)cccc(CNC(c2nnnn2C2CC2)c2ccno2)c1 CCCCC(C)C(=O)N(CCNC(=O)CS(=O)(=O)NCC1CC1)CC C(CNC(=O)C(=O)N(C(=O)CC12COC(C(F)(F)F)(C1)C2)CC)(CC(C)C)OC C(=O)(CCC(=O)c1ccncc1)N(CC(O)CNC(c1ccnn1CCF)=O)C N1(C(c2nc(C)sc2)=O)CCC(O)(C2CCN(C(=O)C=C(Cl)Cl)CC2)CC1 c1(C(N2CCC(O)(C(C)NC(C(C)N(CC)CC)=O)C2)=O)ccn2nccc2c1 O=C(C1=CCCOC1)NCC1CCCCC1C(N1CCOCC2(CC2)C1)=O c1(OC)ncnc(C(N2CCC(N(C)C(C3(C#N)CCCC3)=O)C(C)C2)=O)c1F C1(NC(CN(c2ccccc2)CC)=O)CC12CCN(C(c1cnc(S)[nH]1)=O)CC2 C(=O)(C(F)CC(C)(C)C)N1CCC(C(=O)NCCCCOCC)(OC)C1 C(=O)(C(C)(C)C1=CCN(C(c2ccsn2)=O)C1)NCC(C)Cc1cn[nH]c1 c1(CCCC)ccc(C(C)C(=O)NCc2sc(-c3ccccc3)nc2C)cc1 Cc1n[nH]c(=NCC(CNC(c2c(Cl)cnn2C)=O)C(F)(F)F)o1 N#Cc1ccc(C(=O)NCCC(=O)N2CC(CNC3(CC4CC4)CC3)C2)s1 C1(CNC(C2CCCN(C)C2)=O)CC(C)(C)CN1C(=O)C=CC1CC1 Cc1cc(NC(C2CC(F)CN2C(=O)CN2CCC(C)CC2)=O)cc(Br)c1 CC(CC(=O)NC(c1ccccc1F)CNC(=O)C#CC1CCC1)C(C)(C)C C1(CC(=O)NCC(CC)(CC)NC(c2nnc(S)n2C)=O)CCCCC(=O)N1 C1(C(C)OCc2ccccc2)CCCN(CC(c2cccc(O)c2)O)C1 N1(C(c2n(CCCC)nc(C)c2)=O)CCOCC(CNC(=O)OC(C)(C)C)C1 Cc1cnc(C(=O)NC2C3CC2CN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C3)cc1C c1(C(N(C)CC2(O)CN(C(C3(F)C(C)OCC3)=O)C2)=O)csc2c(F)cccc12 Cc1nc(F)ccc1-c1cc(C(=O)Nc2nccnc2Cl)ccn1 c1(CC)cc(NC(=O)C(C(C)OC)NC(=O)C(C)(COC)CC)cc(O)c1 N1(C(C(CSC)OC)=O)CCC2(CC2NC(c2ccoc2C2CC2)=O)C1 C(=O)(C(O)C1=CCCCC1)NC(C(NOCC(=O)OC)=O)C1CCC1 O=S1(=O)C=C(c2ccc3c(c2)CCC3NCC2CCCCCCO2)CCCC1 C1(CC(=O)NC(C2(O)CCCCC2)C)CCCCN1C(C1(N(C)C)CCC1)=O C=CCC(C(=O)NCc1cc[nH]c1C(=O)NCC(C)CCC)C(C)C C1(NC(C(c2cccs2)SC)=O)C2CC3CN(C(=O)C=C4CCN(C)C4)C1C3C2 n1(C(CC)CC)ccc(C(=O)NCC(C)(O)CNC(c2ccc(C(C)C)[nH]2)=O)n1 N1(C(C(C)OCCCC)=O)CC2(CCC(CNC(=O)CC3COC(C)(C)C3)O2)C1 c1(C(=O)NCC2(C)CCCN(C(C(C)=O)=O)C2)ccc2oc(C)nc2c1 N1(C(c2cnc(OCC)nc2)=O)CCOCC(CNC(=O)CS(C)(=O)=O)C1 CC1(C)CN(C(=O)C2=COCC2)CC1NC(=O)CCCOCc1ccccc1 S(=O)(=O)(c1ccc(NCC2(C)CC=CC2)c2cnccc12)N(C)CC1CCCO1 CC1CCC(C(=O)N(C)C)N(C(c2cccc(NC(=O)NC(N)=O)c2)=O)C1 c1(C(N(CC(C)(C)NC(C(c2nc(C)sc2)=O)=O)C)=O)cnc2ccoc2c1 Cc1ccc(NC(C)C(=O)NC(CO)C(C)NC(=O)C(n2cc(Cl)cn2)C)cc1 C(=O)(C(C)(CCC)CCC)N1CCC(OCC(=O)NC(CC#C)CO)C1 N1(CC)CC2CN(C(C3(C)CN(C(=O)C(F)(F)C4(O)CCC4)C3)=O)CC12 Cc1cnc(N2CC3CN(C(=O)C(F)C4CCOC4)CC3C2)nc1S(C)(=O)=O Cn1ccc(C=CC(N2C(C(=O)NCCCOCCCO)CCC2C2CC2)=O)c1 c1(C(N(CC(CC)NC(=O)CC2CCCOC2)C)=O)ccc2cnccc2c1 C1(C(=O)NCCCCCN(C(c2cc(OC)no2)=O)C)CNC(=O)C(C)(C)C1 c1(OCC)ncc(C(=O)NC2CN(C(=O)C=C3CCCC3)CC2C)cn1 C1(NC(c2csc(CO)n2)=O)COCCN(C(=O)C(O)C2CC2)C1 c1(CNC(=O)NC(c2ccccc2)C2CC2)nc(-c2nc[nH]n2)no1 C(CCC(=O)NC1(CNC(=O)C(C)NC(=O)CC)CCCC1)OCCC C1(CC(=O)NCc2ccns2)CCCN1C(C1CC2(CC2)C1)=O C1(C2CC2)(CC(=O)NCC(C)COC(C)C)CC1 c12ccc(cc1)CC(=O)NCC(C)N(C)C(=O)CC2.c1(CCC)nc(CO)cs1 C1(C(=O)NCC(CNC(COCCC)=O)(C)O)CCc2nc(C)cn2C1 c1(C(=O)NC(CNC(C(C=C)O)=O)C2CCC2)cccc(C(F)(F)F)c1 C(=O)(C(O)CCC(C)C)N1C(C(=O)NCCn2c(C)ncc2)CCCCC1 C1(CNC(CNC(C)=O)=O)CC2(CCN(C(=O)C=C(C)c3cnn(C)c3)C2)CO1 Cc1noc2cc(C(=O)NC3CC3CNC(c3n[nH]c4c3CCCC4)=O)ccc12 c1(CCCCC)nc(C(C)OCC2CCOCC2)n(-c2ccnc(COC)c2)n1 c1(C(N2CC3C(CNC(C4CN(C(C)=O)C4)=O)C3C2)=O)cnc2c(cnn2C)c1 CC1CC(CCNC(=O)C#CCNC(=O)COCC2CCC2)CCO1 c1(NC)cc(C(=O)N(CCCNC(=O)C(C)C(F)F)CCO)cc(Cl)n1 c1(C(=O)NCCCOCCN(C(=O)CC2CSCCS2)C)nccnc1C(N)=O C(=O)(C(C)(C)CC#N)N1CCCC(N2CCN(C(C3(CCC=C)CC3)=O)CC2)C1 c1(C(C)NC(=O)NC(c2noc(C3CC3)n2)C)cc(C(F)F)no1 Cc1ccc(-n2cc(C(N)C3CC3)nn2)nc1.C(=O)(NC)O c1(CC)cc(C(=O)NC2CC3CC2N(C(C24CCC(OC)C2C4)=O)C3)cc(O)n1 C1(C2CCN(C(c3ccn(CCF)n3)=O)CC2)(NC(C2CC(OC)C2)=O)CCC1 N#CCCCCC(=O)NCC1CC1CNC(=O)CCC(=O)NCc1ccccc1 C1(NC(C2(C)CC=CCC2)=O)CCN(C(c2ccc(O)c(N)n2)=O)CC1F C1CCCC(F)(F)C1.C1(CN(C)C)CN(C(C2(C(=O)N(C)C)CC2)=O)C1 CCCC(C)(CCC)C(=O)NC(CC1CC1)C(=O)NC(c1cccc(O)c1)C N1(C(c2c(OCC=C)cccn2)=O)CCCCC(NC(=O)CCCC(=O)OC)C1 N1(C(C=Cc2cn(C)nn2)=O)CCC(C2CCCN(C(c3ccoc3)=O)C2)CC1 C1(C(C)C)CC(C(=O)N(C)Cc2cn(-c3ccccc3Cl)nn2)CCO1 c1(C(=O)NCCN(C(=O)CC2(COC)CC2)CC)ccc(C(C)C)nc1C N1(c2nc(C)cc(OC)n2)CC(NC(=O)CN2CCCCC2C)C2CCCCC12 C(=O)(CCOC1CN(C(c2ccsc2)=O)C1)NCC(C)OC1CCC1 C1(C)(CC)C=C(C(=O)N2CC3CCC3(CC(N3CC(C)C3(C)C)=O)C2)C1 c1(C(=O)NC(C)Cn2cc(C3(C(=O)O)CCC3)nn2)c(F)cc(C#N)cc1Br c1(C(N2CCCC2CNC(=O)NCCN2CCCCCC2)C)c(F)cccc1Br N1(C(c2cc(OC)cc(O)c2)C(=O)NCCC2CC2)CCCC2(CCNC2=O)C1 N1(C(C2CC3CC3N2C(C2CN3CCC2C3)=O)=O)CC=CC12CCOCC2 C1(C(=O)NCCN(C(C2CC23CC3)=O)CC)OCCC1SCCN(C)C C1(NC(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC2CSCCO2)CC1(C)C C1(CC)CCN(C(c2ncn(C)c2C)=O)C1C(=O)NCCCn1cccn1 c1(OCCC)cccc(CN2CC(NC(c3ccc(C(F)(F)F)[nH]3)=O)C(F)C2)c1 c1(C(=O)NCC(C)NC(CN(C)CC)=O)ncc2[nH]ncc2n1 n1(Cc2cc(C)no2)nnc(CC2CN(C(C)C)C2)c1C.c12cn(nn1)C1CC21 c1(C(N2C(C(=O)O)CSCC2)=O)sc2sccc2c1Cl N1(CC(=O)NC2(CN(C(c3cnc(OC)s3)=O)C)CC2)CCCCCC1=O Cc1nc(CC(C)C)oc1C(=O)N(C(C)CCNC(=O)CNC(N)=O)C N1(C(CC2(OC)CCC2)=O)CC2CC1CN(C(c1c(C)ccc(F)c1O)=O)C2 C(=O)(CN=c1ccc(Cl)n[nH]1)N1CCN(C(C2CCCC3(CCC3)C2)=O)CC1 C1(NC(c2cc(OC)ncc2)=O)CCCCCN(C(=O)C(C2CCCCC2)=O)C1 C1(C(=O)NC23C(CN(C(c4cc(C)no4)=O)C2)CCC3)CN2CCCCC2CO1 C1(C#N)(C(N(CCCN(C(=O)C(C)(C)c2cnco2)C)C)=O)CC2CCC1CC2 c1(CCC)cccc(C(N2CCCC(Nc3cnc(OC)nc3)C2)=O)c1 c1(OC)ccc(C)cc1C=CC(=O)N(C(C)CCNC(C1CCC(=O)NC1)=O)C C12(C(=O)NCC3CN(C(CC4(C)CCC4)=O)CC3O)CCC(C)(CC1)OC2(C)C CCCCC(O)CC(=O)NCCN1CCCN(C(c2cc3scnc3[nH]2)=O)CC1 CC1CCC(S(=O)(=O)NCc2nccn2-c2cccc(F)c2)C1 c1(OC)cc(C(N2CCCC(NC(C3CC(C)CO3)=O)C2C)=O)ccc1C CN1CCC(C#N)(C(=O)N(C2CC(NC(=O)C(C)(F)F)C2)C)CC1 C1(C(=O)Nc2c(C(=O)NCC(CC)NC(C)=O)cccc2)CC2CC1CC2=O c1(C(=O)NC2C(NC(C3(C)C(C)(C)C3(C)C)=O)C2)c[nH]c(=O)c2ccncc12 c1(CCNC2(CC(F)F)CCC2)cc(CO)ccc1O CCC(C)(C)C(O)C(=O)NCC1(CNC(c2cc(CO)[nH]n2)=O)CC(F)(F)C1 CC(N)C(=O)NNC(=O)NCCCc1ncco1 Cc1ccc(SC(C)C(=O)NC2CCC(NC(c3c[nH]cc3C)=O)C2)cc1 C(=O)(C#CC1CCOC1)N1CCN(C(CN(C2CC2)CC)=O)CC1CC1CC1 N1(C(CC)=O)Cc2ccccc2C(CNC(c2cnc(O)n2C)=O)C1 N1(C(C=CC(C)NC(C(CCC)CC)=O)=O)CCCC12CCOCC2 C1(CCNC(c2cnc(C(C)C)[nH]2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC(C)O1 C(=O)(CCCCC(C)(C)C)NC1(CCNC(c2n(CC)ncc2)=O)CCCC1 C1(C(=O)Nc2ccc(C#C)nc2)CCCCCCN1C(=O)CC1CCCOC1 N1(C(C(N2CCOCC2)C)=O)CCOC(CNC(=O)COc2cccc(F)c2)C1 C=CCCC(F)(F)C(=O)NC(CCC)CCCNC(c1[nH]nnc1C1CC1)=O c1(C(=O)NC(CNC(c2[nH]nc(OC)c2Cl)=O)C)ccc(C)c(F)c1Br c1(C(=O)Nc2cccc(NC(CCSCC)=O)c2)nccc2c(C)cccc12 N1(c2nnc(CCOC)s2)CC(NC(c2ccc(SC)cc2Cl)=O)CC2(CC2)C1 c1(C(=O)NC(C(C)C)CNC(C2C3(CC3)C23CC3)=O)cc([N+](=O)[O-])ccc1Cl N1(C(CCCOC)=O)CCN(C(=O)CCOCC2CCC2)C(CC(F)F)C1 c1(OCC(=O)N(CC(C)NC(CSCC#C)=O)CC)ccc(F)nc1 C1(C(=O)NC2(C)CC(C(N(CCC#C)CCO)=O)C2)COC(=O)N1C C1(CNC(C(CC)OC)=O)CC2CCCCC2N1C(=O)CCOC1CCCCC1 C12(CC(N3CCCC(COC)C3)=O)CC3CC(CC(C3)C1)C2 Cn1nc(C(=O)NCC(C2CC2)NC(c2c(Cl)n[nH]c2C2CC2)=O)cc1C1CC1 c1(C(=O)NCc2oc(C)c(C(=O)O)n2)cc2c(s1)CCC2=O CCC(C)(CCNC(=O)C(C1CCCCC1)F)NC(=O)Cn1cnnn1 C(=O)(C1=C(C2CCN(CC)C2)N(C2CCOC2)C(=S)NC1c1cnn[nH]1)OC c1(C(=O)NCCOC2CN(C(CC3(C)CCOC3)=O)C2)cnn2c1OCC(F)C2 c1(C(=O)OCC)cc(NC(C(c2nc(Br)cn2C)N2CCC(=CF)C2)=O)ccc1F C1(C(=O)NC(C2(O)CCN(C(c3cnc(N)cn3)=O)C2)C)Cc2ccccc2O1 C1(CC(=O)NCC2CCC2NC(c2cncn2-c2ccccc2)=O)CCCCC1 CCCC(C(=O)OC)C(=O)NC1(CC=CC(N2CCC(F)(F)C(C)C2)=O)CCC1 c1(C(=O)NCC2N(C(CC3OCC(C)(C)C3)=O)CC(O)C2)cnc(S(C)(=O)=O)s1 O=C(CC1CC(=O)c2ccccc21)NCC1CC1NC(c1ccc(Br)cn1)=O c1(CC(=O)NC2(CNC(C3CC(F)C(=O)N3)=O)CC2)c(F)cncc1Cl C1(C(=O)NCC(CCNC(=O)Cc2ccon2)O)CC(c2ccccc2)=NO1 N1(C(c2c(OC)c(Cl)ncc2)=O)CC2CN(C(=O)CN(C3CCC3)C)CC2C1 N1(C(CC(CC)c2ccccc2)=O)CCN(C(=O)CC2CN(CC)C2)CC1CF C(=O)(CCC(C)(C)F)NCC(C)NC(=O)C(c1ccccc1)N(C)C c1(C(N2CCC(F)(CNC(C3CS(=O)(=O)C3)=O)C2)=O)cnc2[nH]cnc2c1 Cc1cn(CC(N2CCCOC(CNC(=O)CC34CC(C3)C4)C2)=O)c(=O)nc1O C(=O)(C1=CCSC1)N(C)CCOCCCNC(=O)C(=O)NCC(N1CCCCC1)=O C1(N(C(=O)CCc2cnco2)CC)CCCN(C(=O)CCc2cccnc2)C1 Cc1nn(C)c(C(=O)NC2COC3(CO)CC2C3)c1Cl.C1(C(=O)N)CCCN1C1CC1 CC1CN(C(=O)CCc2nccs2)CC(C)N(C(c2ccc(C3CC3)nc2)=O)C1 C(=O)(C(C)(C)CC(=O)N1CCC(CN(C)C(c2nccc(F)c2Cl)=O)C1)OC c1(C(N(C)CCN(C(=O)C(=Cc2ccccc2)C#N)C)=O)nnc(O)cc1O c1(OC)cccc(CC(N2CCCC2CN(C)C(c2cc(N)ccn2)=O)=O)c1 C(C(=O)N1CCC(C(N2CC3CC3(CO)C2)=O)(CC)C1)(C(C)C)SCC c1(C(=O)NCC(C)N(C(CNC(CCNC(C)=O)=O)=O)C)cnc(N(C)C)cn1 N1(C(C=C(C)C2CC2)=O)CCOC(CCNC(C2CCN(C)C2)=O)C1 N1(C(C2CCc3n[nH]cc3N2)=O)CCc2ccc3ccccc3c2C1 N1(C(C(=O)NCCC2C=CCOC2)=O)CCOCC1CC1CC1 C=CCC(CN)C(=O)n1c2nnc1s2.C(C)(C)(C)OC(=O)NC C(=O)(C(F)C(C)C)NCCCN(C(=O)CC1CCC2CC12)CC c1(C(N(CCN(C(C2C(OCC)C2)=O)C)C)=O)csc(-c2ccccc2)n1 C12(C(=O)OC)CCCCC1(C(=O)N(C(c1ccco1)C1CC1)C1CC1)CC2.CC CCC(C)CCCC(=O)N1CCOCC1CNC(=O)CCCC(N)=O CCCC(CC(C)C)C(=O)NC1(C)CCCCC1C(=O)Nc1ccc(O)cc1CC C(=O)(C1c2c(Br)cnn2CCN1Cc1nc(C)c2n1CCC2)OC C#Cc1cncc(C(=O)NC(C)C(C2CC2)NC(=O)CCc2ccccc2)c1 C1(C(=O)NCC2CC(NC(c3c(CC)n(C)nc3)=O)C2)Cc2nncn2C1 C(=O)(CC(C)(C)C(F)F)NC(C)CNC(c1ccc(F)cc1)=O C(=O)(N(O)C(C)C)c1c(CCC)nco1 c1(OCC)ccc(-c2cnc(NC(c3cc(Cl)cc(I)c3)=O)nc2)c([N+](=O)[O-])c1 CC(C)(O)C(F)C(=O)NCCC(=O)NCCS(C)(=N)=O C1(n2cc(C(CC)(O)CC)nn2)CCC(C(=O)NCC2CC2(C)C)CC1 CC1CC(C(N2CC=CC2(C)C)=O)CN1C(=O)Cc1ccco1 Cc1ncc(C(=O)NCC2(F)CCN(C(=O)CN3CC(=O)NC3=O)C2)n1C c1(C(C(=O)NN2CCOCC2)N(CC(C)(C)CO)C)cn(C)c(=O)c2cccnc12 CC1CC(NC(=O)CCOc2ccc(F)cc2)CN(C(c2ccncc2F)=O)C1 OCC1(c2ccccc2)CCC(NCCCOC2CCOC2)CC1 C(C(CO)(CO)NC(=O)C=CC=Cc1ccccc1)N(C)C(C1CCC2CC12)=O C1(NC(c2c(C)n(C)nc2)=O)CC1C1CCN(C(C2CCOC(C)C2)=O)CC1 c1(NC)ccc(F)cc1C(=O)NC(CNC(=O)C(C)=C1CCC1)C(C)C N1(C(c2occ(C)c2C)=O)CCCC(CNC(c2cccc(C(N)=O)n2)=O)CC1 c1(C(=O)NCC2CN(C(C3(CC(C)=O)CC3)=O)CC2C)cc(F)c(F)cc1F C(CC(C(C)C)NC(c1csc(CO)n1)=O)N(C(c1c(C)snn1)=O)C C(=O)(C(=O)CC(C)C)N(C(C)C(=O)NCC1CC1(C)C)CC c1(C(=O)NCCC2(CNC(C3C(CC)C3)=O)CC2)cc2n(n1)CCCC2O CCCCC(O)C(C)C(=O)N1CC(F)(F)CC1CNC(c1cnc(CC)[nH]1)=O N1(C(C2(C(C)(C)C)CCCC2)=O)CC2CN(C(C3CCCO3)=O)CC2(C)C1 Cc1cc(C(N2CC(CC(C)NC(c3cc(CO)[nH]n3)=O)C2)=O)c(F)cc1Cl C(CCCC(=O)N(CCCN(C)C(c1scnc1C)=O)C)OCC c1(CCN2CCC(CNC(C(CCC)OCC)=O)C2)ccc(Cl)nc1C c1(C(N(CCN(C(C23C(C)OC(CC2)C3)=O)C)C)=O)ccc2cccc(F)c2n1 CCCCC(C(=O)NCC1(F)CCN(c2cc(OCC)ncn2)CC1)C(C)C C1(N(C)C)CCC(C(=O)NCC2CCCC2NC(=O)C=CC(C)(C)C)CC1 N1(C(c2sc(C)c(Br)n2)=O)CC(NC(C2CCOC2)=O)CC1(C)C Cc1nc(C)c(C(=O)NC2(CO)CN(C(c3ccnnc3Cl)=O)C2)c(C)n1 N1(C(C(C(C)C)CO)=O)CC(C)OC2(CCN(C(=O)CC3CC(C)(C)CO3)C2)C1 C1(NC(C(=O)NC(C)C)=O)CCC2CCC1CN2C(=O)CC1CN(C)C1 c1(C(=O)OCc2c(C)onc2)cc(C(=O)NCc2ccc(F)cc2)ccc1Br C1(NC(C2CCN(c3nccc(Br)c3F)C2)=O)CC[Si]2(CCCC2)CC1 c1(C(N2CCCC(CCNC(C3COC(=O)O3)=O)C2)=O)ccc(Cl)nc1O N1(C(c2c(=O)ccn(C)c2)=O)CC2CCC(NC(C3CCC(=O)NC3)=O)C2C1 c1(OC)ccc2c(CCNC(N3CCCC3c3cccnc3)=O)c[nH]c2c1 C1(CC)CC(C(N2CCC(C(C)(C)NC(=O)CCC(C)SC)C2)=O)CCO1 N1(C(CC2(NC(C)=O)CC2)=O)CCC(CCC(C)(C)NC(=O)C(O)C(C)C)CC1 C(CNC(c1cccc(O)n1)=O)(CC(F)(F)F)NC(c1cncc(OCC)c1)=O c1(C(N2CCC2CNC(C2(F)CC=CCC2)=O)=O)cc(-n2cccn2)ccn1 c1(CNC(C(CN(C)C)NC(COCCC=C)=O)=O)ncc[nH]c1=O C1(CCC(=O)N(CC(C)O)CC(C)O)CCCN(C(c2cn[nH]c2)=O)C1 CN1CC(CNC(=O)C(O)C2(O)CNC2)C(F)(F)C1 C1(C(=O)NCCCN(C(C2C(CCC)C2)=O)C(C)C)CS(=O)(=O)CC(=O)N1 CCC(O)C(C)(C)C(=O)N1CCC1CNC(c1c(-c2ccsc2)c[nH]c1C)=O N1(C(c2ccc(C)n2C)=O)CCC(NC(C23C=CC(CC2)C3)=O)C(O)C1 c1(OCCCCC)ccc(C(=O)NC2CC(NC(C3(C)CC3(C)C)=O)C2)cc1 C#CCCCCCC(=O)NC1CCC1CNC(=O)Cc1cnccc1OC C1(C(N2CCC(C(=O)OC)C2C)=O)CC2CN(C(=O)CC3CCCCO3)CC2C1 C(N=c1nc(N2C3CCC2CC3)c2c([nH]1)CSC2)C1CC=CCC1 S(=O)(=O)(C(F)(F)F)NC(=O)CC1(CO)CC1.C1(CC)(N)COC1 C(c1ccc2c(c1)OCO2)=CC(N1C2C(NC(Cn3c(C)ccn3)=O)C(C2)C1)=O c1(C(c2nnnn2C2COC2)NCCCCOCCO)ccc(F)cc1 c1(C(N2CCC(N(C(C(CC=C)C(C)C)=O)C)C2)=O)cc(F)cc2cc[nH]c12 c1(NC(C=CCN(C)C(c2cccnc2C2CC2)=O)=O)c(CO)cnn1C c1(CC(=O)NC2CC(F)(CNC(C(C)=C3CCC3)=O)C2)ccc(C)c(Cl)c1 c1(NC(C2CC(C)N(C(=O)CCCCCF)C2)=O)ccn2nccc2c1 C1(=CC(=O)NC2C(CNC(=O)CC3CCCCC3)COC2)CN2CCC1CC2 c1(OCC(N2CC(C)C(NC(=O)CC3CC4(CC4)CO3)C2)=O)ccc(Cl)cc1Cl N1(C(=O)NC2CCC(CC(N)=O)C2)CC2(CCC2)C12CCC2 C1(NC(c2n(C=C)ncc2)=O)CN(C(c2cc3sccc3[nH]2)=O)C(C)(COC)C1 C(=O)(CP(C)(C)=O)NCCN(CCOC)C(c1cnc(COC)nc1)=O C=CCCCCCC(=O)N1CC(NC(c2coc(Cl)c2)=O)CC1(C)CC C1(C)(C(N2CC(OC)(CNC(=O)C(C)CCN(C)C)C2)=O)C(C)(C)C1(C)C CC1(C)CCCN(C(c2ccco2)=O)C1C(=O)NC(c1cccc(O)c1)CCO c1(C(C)NC(Cc2cc(OC)c(Br)cc2)=O)cn2c(n1)CCCC2 Cc1c(NC(C2CCCN(C(=O)C(C)CO)C2)=O)cccc1[N+](=O)[O-] CC1=NOC2(C1)CC(c1nc(-c3ccccn3)nn1C1CCN(C(C)(C)C)C1)C2 C1(C(N)=O)C2CCC(C2)C1NC(c1ncccc1NC(C1CCCCCC1)=O)=O C(C(C)(O)C(=O)N1CC(C)(NC(c2cc(-c3cccs3)[nH]n2)=O)C1)OC C1(C2CCN(C(CCCC)=O)C2)CCCCN1C(=O)CCNS(C)(=O)=O N1(C(C2(CC#C)CCCO2)=O)CC2(CCNC(C3CC3C(N)=O)=O)CCC1CC2 N1(C(COC2CC(NC(c3c(C)non3)=O)C2)=O)CC2(CCC2)C1 C(=O)(CCCC(=O)N(C1CCCN(C(=O)COc2cccnc2)C1)C)OC C1(C(=O)NC2(c3cn(-c4n(C)ccn4)nn3)CCCC2)C(C2CC2)C1(F)F c1(N2C(C)CC(NC(C34C(C)OC(C)(C3)C4)=O)C2)nc(Cl)nc2c1cnn2C C1(CNC(c2cc(OC)ns2)=O)CCN(C(=O)C(C)=CC(C)(C)C)C(C)C1 C(N=c1ccnc(-c2ccccc2)[nH]1)C1CC(NC(=O)Cc2cccs2)C1 C1(C)(c2c(OC)cccc2)CCN(C(=O)CN2CCC(F)(F)CC2)CC1 CC(CC(=O)N1CC(C(O)C(N2C3COCC2C3)=O)C1)P(C)(C)=O N1(C(C(=O)NCC(=O)N(c2ccsc2)CC)C2CC2)CCOCC1 N1(C(c2ccc(CO)o2)C(=O)NCC(=C)C)CC(c2ccccc2)C(C)(C)C1 Cc1c(CS(=O)CC(C)C(C)C)cnn1C c1(CC)nc(C(=O)NC2CC(NC(c3cnc(NC4CCC4)nc3)=O)C2)c(C)o1 C(=O)(C(CC)CCOC)NCC(=O)N(CC(COC)(C)C)CCC=C C#CC1(CNC(=O)C(C)(CO)NC(=O)COCC2CCCC2)CCCC1 C(=O)(CC(C=C)CCC)N1CCC(C(C(=O)N(CC#C)CC2CC2)C)CC1 CCC(CNC(=O)Cn1ccnc1)(CC)C(=O)N(C)CC12CCC(CC1)C2 CN1CCN(C2(C(N3CCCCC3CNC(c3ncc(C(=O)O)s3)=O)=O)CC2)CC1 c1(C(=O)NCC2C(C)CN(C(=O)Cc3ccc(Cl)s3)CC2)ccc(F)c(C#N)c1 C(C)(C)(CC(=O)NCCc1cn(C)nn1)NC(COCC#C)=O C1(NC(=O)CCc2ccc(F)cc2)CCCC12CCN(C(C13CC(CO1)C3)=O)C2 c1(CC)nc(C)[nH]c1C(=O)NC(C)CN(C(=O)CC1CCCO1)C c1(C(=O)NCC(C)CNC(=O)CC2COC3CC2C3)ccc(F)cc1C(F)F C1(C(N2CC(NC(c3n(CC)ccn3)=O)C(C)C2)=O)CCc2ncnc(C)c2C1 C1(CC=C)(NC(=O)CCCCCO)CCCN(C(=O)Cc2ncccc2C)C1 n1(CC2CCC(NC(N3CCC(C4N=N4)CC3)=O)C2)cnc2ccccc12 N1(C(C2C(C)C(=O)C2)=O)CCN(C(=O)C=Cc2cccc(CO)c2)CC1C CC1(C)OCC2CC12C(N1CCCCC1CNC(C1(n2cncn2)CC1)=O)=O C(=O)(C(C)C(C)C1CCCCC1)NC1(F)CC(N(CCCCN(C)C)C(C)=O)C1 N1(C(c2scc(C(C)C)n2)=O)CC2CCC1CN2C(c1csc(Br)n1)=O N1(C(CCNC(C)=O)=O)CCC(C)(C)C1CC(=O)NCCC1CCCC12CC2 C1(NC(CCSC)=O)CC2CCC1CN(C(C13CC(CO)(C1)OC3C)=O)C2 c1(C(=O)OC)ccc2[nH]c(=NC(C)CCSC)oc2c1 Cn1cc(C#N)cc1C(N1CCC(CCNC(c2c(Cl)nsc2Cl)=O)C1)=O C(N=c1[nH]nc(CC(C)C)s1)C1OCCN(C(C(=Cc2cn[nH]c2)C)=O)C1 Cc1cn2c(n1)CCC(C(=O)NC1(c3ccc(Br)cc3F)CC1)C2 c1(C(N2C(CCC)CN(C(=O)C(C)(C)N(C)C)CC2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(NC(C(CC)CCOC)=O)CN(C(C2(C)CC=CCO2)=O)CC2(CCC2)C1 C(=O)(C(O)CCCNC(=O)CCn1cncn1)N(C1CCN(CC)C1)C CC1=NC(C)(COC(=O)CCCN(C(=O)COc2ccccc2)C)CS1 CC(C)CS(=O)(=O)CC(=O)N1CCCC1CNC(=O)CSc1cccc(O)c1 N1(C(c2nc(C)[nH]n2)=O)CC(NC(=O)C2CC2)C(C(F)(F)F)C1 c1(C(=O)NC(C2CCOC2)CNC(c2cnc(C)o2)=O)c(C)nn(C)c1C(F)F C1(CN(C(=O)NCc2n(CC)ccn2)CCO)CCC(C(F)(F)F)CC1 C1(NC(C(C)NC=O)=O)CCCC(CNC(=O)CN2CCS(=O)CC2)C1 C(C(C)(C)CCNC(c1ccc(C)n1C)=O)NC(C(C1CC(F)(F)C1)OC)=O c1(CN(C)CC2(CO)CC=CC2)ccc(OC)c(Oc2ccccc2)c1 CC(=O)CCCC(=O)N1CCN(C(c2ccnn(C)c2=O)=O)CC1CS(C)(=O)=O c1(-c2c(F)ccc(NC(c3c(OC)ccc(C)c3)=O)n2)ccc2occc2c1 N(C1COc2c(F)cccc21)C(c1ccc(Cn2cc(COC)nn2)o1)=O C12(NC(C(C3CC3)SC)=O)CC(CO)(C1)OC21CN(C(c2ccn(C)n2)=O)C1 C1(C(=O)NC(CC)C2CC2)CCN(C(=O)CCc2ccn(C)c2)CC1O C(=O)(C(C(=O)NC1CCN(C(c2c[nH]c(C)c2)=O)CC1C)C(C)C)OCC c1(OC)cnc(Br)c(NC(=O)CC2C=CC(NC(c3ccc(F)cc3)=O)C2)c1 N1(C(C)C)CCOC(C(=O)NCC(O)CNC(c2ccccc2C2CCC2)=O)C1 c1(C(N(C(CNC(c2c(C)snn2)=O)C)C)=O)ccc2c(c1)CC(=O)NC2 N1(C(C=CC(CC)C)=O)CC(NC(=O)CC(C)(C)C)CC12CCOCC2 C1(CNC(C(C=C)O)=O)Cc2ccccc2CN1C(c1cc(F)cnc1O)=O c1(C(N2CCC(C(=O)NCC(c3ccc(C)cc3)O)C2)=O)c(C)nn(C)c1Cl C(=O)(CC1=CCCCC1)NC(C)CC(=O)NCc1c(O)cccc1F N1(C(c2c(C)csc2Cl)=O)CC(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)C1 C1(C(=O)NCCN(C(=O)C(CCSC)N(C)C)CCSC)(CC)CCNC1=O C1(N2CC(CN(C)C)OCC2)CC2(C1)CN(C(=O)C=CC(N1CCOCC1)=O)C2 c1(C(N2C(CNC(=O)C=CC(F)F)CCC2)=O)ccncc1Cl c1(NC2OCCN(C(=O)Nc3c(CN)cccc3)C2)ccc2ncccc2c1 Cc1cc(C(=O)NC(C2CN(C(=O)C(C)OCCC(C)C)C2)C)cc(C)c1 c1(C(=O)NC(CC)CO)cc(O)nc2c1CN(C(C1(O)CC1)=O)CC2 c1(C(=O)NC2(CCNC(=O)COCCc3ccccc3)CCC2)ccc(O)nn1 c1(C(N2CCOCC(CNC(CCOC(C)C)=O)C2)=O)cc2ccncc2[nH]1 c1(C(=O)NC(CNC(Cc2cc(C)no2)=O)(C)CC(C)C)cc2c[nH]cnc-2n1 N1(C(C(COC)C)=O)CCC(NC(=O)C(=Cc2cnn(C)c2)C)C12CCCC2 C1(C(N(CC(=O)NCC2(C)CCC(=O)N2)CCOC)=O)CCN(C)C(C)C1 c1(CC)cc2c(CC(=O)NC3CC(CNC(=O)CC4CC45CC5)C3)csc2s1 c1(CC)cc(C(N2CCC(C(CO)N(CCC#N)C(C)=O)CC2)=O)n(C)n1 C(=O)(CCCC(=O)NCC(C1CC1)NC(=O)CCc1ccc(Cl)s1)NCC c1(C(C)C(=O)NCC(C)(C)CNC(=O)CCC2CC2C)ccc(F)c(F)c1 c1(C(=O)NC(CC(C)NC(c2cc(CCOC)on2)=O)C)cnc2n1CCOC2 C1(C(N(CC(C(C)C)OC)C)=O)CCCN(C(C2CSCC(=O)N2)=O)C1 C1(NC(C(C)(C)CO)=O)C2CC3C(C2)C13C(N1CCNC(=O)C1CCO)=O C1(CC)(NC(=O)CCc2ccn(C)c2)CCOCC1.C12(CCCC1)C(=O)N2 C1(CCCNC(c2cncn2C2CC2)=O)CCN(C(=O)CC2CCC2(F)F)CC1 C(=O)(CN=S(C)(C)=O)N(C(c1ccncc1)CNC(=O)CNc1ccccc1)C C(=O)(C(CC(C)C)C(C)C)N1CC(OC)(CNC(=O)Cc2cccn2C)C1 C(=O)(CCCC(C)C)NC1CCN(C(C(C)OCc2cccc(C)c2)=O)C1 c1(C(CCC)NC(C2CN(C(=O)CC)C2)=O)cc2c(s1)CCC2 c1(OC)ccc(C(N2CCCC2n2cc(C(C)O)nn2)=O)c(C2CC2)c1 c1(OCC(=O)N(C2CCC(NC(C3(C)CC3(F)Cl)=O)CC2)C)ccc(F)cc1 c1(-c2onc(C(CC)Cc3ccccc3)n2)cc(C(=O)OC)cn1C CC1CC=CCC1NC(=O)C(C1(O)CCC1)NC(=O)C=CC(F)(F)F CCCCCCC(C)C(=O)NC(Cc1ccccc1)CCOC(F)(F)F C1(CC(N2C(CN(C(C(CCSC)O)=O)C)CCC2)=O)CCC(=O)NC1=O c1(C(=O)NCC2C(NC(c3cnc(C(=O)OC)s3)=O)CCC2)ccc(C)cn1 CCC(CC(=O)NC1CN(C(C2CCC=CCCC2)=O)C2(CCC2)C1)CC(C)C c1(OC)ncc(Cl)cc1C(=O)NCC(C)CNC(C1CC(N2CCOCC2)C1)=O C1(C)(NC(c2c(C)coc2)=O)CCCN(C(c2cc(C)c(Cl)cn2)=O)C1 C12(NC(c3cnc(SC)n3C)=O)CC3CCC(C1C2)N3C(C1(C)CCC1)=O Cc1cn2cccc(NC(C3CC4CCN(C(=O)CCNC(N)=O)CC34)=O)c2n1 c1(NC(C2c3nc(oc3)C3N2CC3)=O)ccccn1.C1(C)(CCO)CC1.CS c1(C(=O)NCCNC(c2c(C)noc2C)=O)ccc2c(ccn2C)c1 c1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)C2)cn2c(Br)c(C)nc2s1 N1(C(c2scc(C(N)=O)c2)=O)CCC(CNC(=O)C(F)=CCCF)CC1 Cc1scc(C(N2CCOC(CNC(C3C(C)(C)C3(C)C)=O)C2)=O)c1C1CC1 Cc1cc(C(=O)NCCC(C)N(C2CCCCC2)C(C2(CCF)CCC2)=O)n(C)n1 c1(C(=O)NCC2N(C(CC(=C)C)=O)CC(F)(F)C2)c(C)cc(C#N)cc1C C1(N(C(C=CC)=O)C)CCCC(N(C)C(c2cnc(-c3cccs3)o2)=O)C1 C1(COC)(NC(=O)Cc2nc(C3CCCC3)no2)CCCNC1 c1(C(c2n(CC)nnn2)NCc2ncoc2CC)cnn(C)c1C(F)F C=CCC(C)(CC)C(=O)N(C)Cc1cn(CCCC2CC(F)(F)C2)nn1.OC N1(C(C2(CCC=C)CN(C(=O)C(C)(C)C(C)C)C2)=O)CCN(C)CC(C)C1 c1(OC)ccc(NC(C2(NC(=O)C(F)OC(F)(F)F)COC2)=O)cc1 c1(C(=O)NCCOC2CCN(C(C(C)SC)=O)CC2)ccnc(O)c1Br C1(C(=O)NC2CCCC(F)C2)CC(F)(F)CN1c1nnc(O)s1 Cc1cccc(Br)c1C(=O)NC1CC1NC(=O)CCCOc1ccccc1F CC(C)(CNC(=O)CC1CC1c1ccccc1Cl)C(=O)O.c12cn(nn1)C2 c1(C(C)C(=O)NC2CC(CNC(C3CCC(C)O3)=O)C2)ccc(Cl)c(Cl)c1 C(=O)(C1=NOC(CNC(=O)CC2(C)CC2)C1)N(C1(CCO)CC1)C C12CN(C)CCN1C2=O.C12(CNC(c3ccc(OC)s3)=O)CC1COC2(C)C c1(C(=O)NCC2CN(C(c3ccc(C)nc3C)=O)CC2C)ccc([N+](=O)[O-])cn1 N1(C(C(=O)NC(COC)=O)=O)CCC(N(C(=O)CSCCC(N)=O)C)CC1 C(=O)(C1CCc2c[nH]nc21)N1CC(NC(c2c(N)sc(C)c2C)=O)CC1(C)C CN1CCCCC1C1C2CN(S(=O)(=O)CC#N)CC12 C(N=c1[nH]c(=NCCOCCF)[nH]c2cccc(F)c12)C1C(C)OCC1 C1(C(=O)NCC2CC(NC(C3CC(F)(CO)C3)=O)C2)CCCCCC1(F)F c1(C(=O)NC2(C)CN(C(C3CCn4nnnc4C3)=O)C2)cc2cccc(Cl)c2s1 C1(CNC(c2n(C)nnc2)=O)CN(C(=O)C(=O)CCc2ccsc2)CC(C)(C)O1 O(NC(=O)C(CCC=C)CC#C)C(C#C)CCC.OC N1(C(COCCC=C)=O)Cc2n[nH]cc2C1C(=O)NCCCc1ccn(C)n1 c1(C(=O)NCC2CN(C(C3C(=C)CC3)=O)C(C)C2)ccc(C)c(O)c1 C(C(C)(C)C(=O)NC1CC(c2cn(CC3CCO3)nn2)C1)N(C)C Cn1cc(C(=O)NCCCC2CN(C(c3cc(Cl)n(C)n3)=O)CCO2)n(C)c1=O c1(C(N2CC(NC(C(C)C#N)=O)C(CO)C2)=O)cc2cnccc2o1 c1(C(=O)NC(CNC(C2C(COC)C2)=O)(C)C(C)C)cccn2ncc(Br)c12 c1(CCC(N2CCCCC2c2cn(CCF)nn2)=O)cccc(Br)c1Cl C12(CNC(c3ccns3)=O)CC1CN(C(=O)Cn1ncc(Br)n1)C2 c1(C(=O)OC)cc(C(N2CC(O)CC2CNC(c2[nH]nnc2C)=O)=O)cc(F)c1 Cc1ccc(C(=O)NCC(C)NC(=O)C(c2cccc(Br)c2)(C)C)c(N)c1 C(C1CC(C)Oc2ccccc21)NC(Cc1c(OCC(C)C)cccc1)=O C1(NC(c2cc(C(C)C)on2)=O)CCCN(C(C2CC3(C2)CC(O)C3)=O)C1C C1(CNC(=O)CSc2nnc(S)s2)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O C1(CC(=O)NCC2(C)CCCN2C(c2cc([N+](=O)[O-])c[nH]2)=O)CC(F)(F)C1(F)F C(=O)(C(C)(C)CCC#N)NC.Cc1cc(C)n(CC(=O)NCC23CCC(CC2)C3)n1 Cc1nc(NC2CC(NC(c3ccc4nonc4c3)=O)C2)c2cc(Br)ccc2n1 N1(C(c2ccc(CC)s2)=O)CCCC(C)(C)C1CNC(=O)CN1CCC1C c1(C(N2CC(C(C)NC(C(C=CC)O)=O)C2)=O)csc(C)c1Br c1(CN(C)Cc2cc(-c3ccncc3)no2)ccc(CNC(=O)C(C)(C)CCl)cc1 C(=O)(CC1=CCCCC1)N1CC(CC(C)NC(C2(CNC(N)=O)CC=CC2)=O)C1 C1(C)(C(=O)NC2(COC)CC2)CN(C(=O)C(C(C)C)NC(C)=O)C(C)(C)C1 C(=O)(C(CO)C(F)(F)F)N1C(C)CC1C(N1CC(c2ncccn2)C1)=O C=CCC(CNC(=O)CC1CCN(C(=O)C(C)(F)C(C)(C)F)C1)CC(C)C C(=O)(C(C)(C)CCC(=O)NC1COCC1CNC(C1CN(CC(C)C)C1)=O)OC N1(C(C2(C)CCOC2)=O)CC2(C1)SCCC2NC(c1csc(-c2cnc[nH]2)n1)=O c1(C(=O)NC23CC(C(=O)N(c4ccsc4)CCO)(C2)C3)cc2ccccc2[nH]1 CC1CC(C)N(C(=O)CSC(F)F)CCN1C(=O)C#CC1(C(F)(F)F)CC1 N1(C(c2c(C)csn2)=O)CCCCC(C2CN(C(c3ncn4c3CCC4)=O)C2)C1 C1(CNC(c2c(C)n(C3CC3)nn2)=O)CCC(C)CN1C(=O)CC1(O)CCC1 C1(C(=O)NCC(CC)C#N)(CC)CCCN(C(=O)C=CC2CCC2)C1 C1(CN(C(=O)CC2(CO)CC2)C)CCN(C(c2scnc2C(F)(F)F)=O)CC1 C1(N(C(=O)CC2N(C(C(CC=C)OC)=O)CCC2)C)CCC(C)(C)CC1 C1(NC(c2cc(C(C)C)[nH]n2)=O)COCCN(C(=O)C=Cc2ccsc2)C1 CC1(C)CN(C(C2CCCC(F)C2)=O)CC1NC(C1C2CCC(=O)C12)=O Cc1nccnc1C(C)NC(=O)C(C1CCCN(C(=O)CC2(C)CC2)C1)C C(C(=O)N1CC=CC(NC(=O)Cn2nc(C)oc2=O)C1)(C(C)C)NC(C)=O Cc1cccc(COCC(N)Cc2ccccc2)c1.C1(C)C(=O)N1 C1(C2CCN(C(=O)CCC3CCC(C)O3)CC2)(NC(c2c(C)nn(C)c2)=O)CC1 c1(C2C(C(=O)NCC3CCN(C(c4cc(C(C)C)no4)=O)C3)C2)ccc(F)cc1 N1(C(CS(CC)=O)=O)CCC(C2CC2)(CNC(c2conc2C2CCC2)=O)C1 C1(NC(c2c(C)nc(Cl)cc2)=O)CC2CC1CN(C(=O)Cn1nnc(=O)[nH]1)C2 C(=O)(C(C)(CC#C)NC(=O)C(C)OC1CC1)N(CC#C)CCOC c1(CC(=O)NCC(C2CC2)NC(C2CCN(C)C2)=O)csc2c(F)cccc12 c1(NC(C2(CC)COC2)=O)cccc(NC2=NCCC2)c1 C1(C(=O)NCC2(CCO)CCC2)CC2C=CC1N(CC=Cc1cocn1)C2 C(c1cocn1)=CC(=O)N(CC(C)NC(C1CC2(CC2)C1)=O)C CCCCC(F)C(=O)N1CC2CC1CN2C(=O)CC12CCCC1C2 c1(C(=O)NC(CC(=O)N(C(CC)C)CCO)CC2CC2)nnc(O)nc1O C(C(O)C(=O)NOC(c1ccncc1)C)NC(c1c(CC)cns1)=O c1(C(N2CCN(CC(=O)Nc3nccnc3Br)C(=O)C2)=O)ccc(Br)c(Cl)c1F c1(OC)ccc(C(N2CC(N(C)C(c3nnccc3C)=O)C(O)C2)=O)cc1OC c1(C(N(C(CC)CC(=O)NC2CCCC2OC)C)=O)coc2c1COC2 O=C1C2CCC3(CCC3)CN2C(=O)N1CCSc1cccc(Cl)c1Cl Cc1cnc(CNCCCC2C=CCC2)nc1 N1(C(C2CC(CCC)C2)=O)CCC2(C1)C(=O)N2.C(C(C1CC1)C1CC1)OC n1(CCCC)nccc1C(=O)NCCN(C(=O)CN1CCOCC1)C(C)C C(=O)(N=c1nco[nH]1)NC1(COC)CNCCO1 c1(OC)ccc(CC(CNc2ccccc2NC(=O)C2CC2)CO)cc1F C1(CC(=O)NC2C3CN(C(c4c(CC)nns4)=O)C(C3)C2)CC2(CCCC2)CO1 c1(SC)ncc(N)c(C(=O)NCC2CCCC2NC(c2cc(C)ncn2)=O)n1 C=C(Cl)CC(C(=O)NCC(C)N(C)C1CC1)NC(c1cccs1)=O c1(C(N2CCCC(C)C2)=O)nccc(N)c1Cl.C(=O)(CCC(=O)N(C)C)N(C)C N(C(=NCCC1CC(F)C1)NC1CCC1)C(COC)C C1(NC(CSCC(=O)OC)=O)CC12CCN(C(=O)C(c1ccccc1)=O)CC2 C(=O)(C1CCCc2cccnc21)NC(CNC(CCC(=O)NCCC)=O)C(C)C C(c1ccc(OC)c(OCC)c1)=C(C(=O)NC1CCN(CC=C)CC1)C C1(NC(c2ccccn2)=O)CCC2CCN(C(c3ccc4nsnc4c3)=O)C1C2 CC1C(NC(c2cncc3ccsc23)=O)CC2CCC1N2c1nnc(C2CC2)s1 C1(C(=O)NCC(C)NC(=O)CCC2CC2(C)C)CCCN1N=O Cc1ccc(Br)c(F)c1C(=O)NC1(CNC(C2(C#N)CCC2)=O)COC1 c1(CN2C(C(=O)Nc3c(C(=O)OC)scc3Br)CCC2)c[nH]c2cc(Cl)ccc12 C1(NC(C2(NC(=O)C(F)F)CC(O)C2)=O)CC2(CNC(=O)O2)C1 c1(OCCCC(=O)OC(c2cnn(CCC3(N)CCC3)c2)=O)ccc(F)cc1 c1(-n2c(C(n3cncn3)C)nc(-c3cc[nH]n3)n2)ccc2ncccc2c1 N1(C(C(n2ccc(C)n2)C)=O)CC(NC(C2CC2c2oncc2C)=O)C2(CC2)C1 O=C1Nc2cc(Cl)ccc2N(CC2CN(C(C3CCCC3)=O)CCO2)C1C1CC1 c1(NC2C(CNC(=O)CC3CCCS3(=O)=O)CC2)cc(C(F)F)nc2ncnn12 C(=O)(CCCCC(N)=O)NC(C)CN(C)C(c1cc(-c2ccco2)c[nH]1)=O c1(C(N2CC(C)C(NC(C3CC34CCCCCC4)=O)C2)=O)c(F)ccc(F)c1F C12(NC(C3CC(=C)C3)=O)CC(CNC(c3cc(CO)[nH]n3)=O)(C1)OC2C CC1(C(=O)NCCCC2CCN(C(=O)CCC3CC3(Cl)Cl)CC2)CCC(=O)N1 c1(OC)ccc(NC(C2CC(NC(c3cccc(C)c3)=O)C2(C)C)=O)cc1C c1(C(=O)NCCC(C)N(C(C(C=C)c2ccccc2)=O)C)ccccc1C(C)C N1(C(c2cc(CNC(CCOC)=O)oc2)=O)CC2CC1CN2Cc1ccccc1 C(=O)(C(C)(C)CC#C)N(CCC(C)NC(c1nc(C#C)sc1)=O)C CC1OCCCC1C(=O)NCCCN(C(=O)CCOC1CCCC1)C C12(NC(c3n(CC)c(O)nc3)=O)CCC(C1)N(C(=O)COC1CCC1)C2 CC(CC(=O)NC12CC(C(=O)N(C3C4CC5C(C4)C35)CCO)(C1)C2)CC(F)(F)F c1(CC)ccccc1C(=O)NCC(C(C)C)NC(=O)CNS(=O)(=O)CC c1(C(=O)NC2CC(C)(NC(C(CCCC)C)=O)C2)ccc(OC)c(F)c1N c1(CN2C(C(N3CCCCC3CCO)=O)CC(C)C2)cc2cc(Br)ccc2[nH]1 O=S(=O)(c1ccc(NC2CSc3ccccc32)c(Br)c1)NCc1cc(Cl)sc1Cl C(=O)(CCCCCCc1cn(CC2CCCC2)nn1)N(C1CCCC(C)C1)CCF NS(=O)(=O)c1ccc(C(=O)NCC(CO)NC(=O)C(O)c2cnc[nH]2)o1 N1(C(C(C)OCCCC)=O)CCCC(C)(NC(c2ccc(=O)n(C)n2)=O)C1 C(=O)(C1CCCNc2ccccc21)NC(C1CCN(c2ncc(C)c(O)n2)C1)C c1(C(=O)NCC(CNC(=O)C=C2CC2)O)n[nH]cc1C1CCC1 c1(C2(CN(C(=O)CCC3CC3)C3CN(C(=O)C4CC4)C3)CC2)ccc(F)cc1Cl N1(C(CCC=C)=O)CC(CC(=O)N(C)CCN2CCCC2)C2(CC2)C1 c1(C(=O)NC2CCC(NC(C(C)OCC)=O)CC2)c(C)[nH]c2ccc(Cl)cc12 Cc1cc(C(=O)N(CC(O)CNC(=O)C=C(Cl)Cl)C)ncc1Br N1(C(c2n(CC#C)ccc2)=O)C(C)CN(C(=O)C=C(Cl)Cl)CC1C N1(C(C2C(C)(C)CO2)=O)CC(CO)C2(C1)CN(C(c1cncc(Cl)c1Cl)=O)C2 c1(CC(C)(C)C)ccc(C(=O)NCCC(O)CNC(=O)C(CO)N(C)C)cc1 c1(CS(C)(=O)=O)nc(C(=O)NCC2CCN2C(c2cc[nH]n2)=O)cs1 C(C(=O)NC1(C)CN(C(c2cn(CC(N)=O)nn2)=O)C1)(C(C)C)SC N1(Cc2cccc(OC)c2C)CCOC2CC(C(=O)O)CCC12 c1(C(=O)NC(CCC)CNC(=O)C(CC)NC(N)=O)cc(C)n(C)c1C C=CC1(NC(C2CCCN(C(c3cn(C)cn3)=O)C2C)=O)CCCCC1 C1(CCC)CN(C(c2c(Cl)c(CC)nn2C)=O)CCN1C(=O)CCSC C12CCN(CC1)C(=O)C1(CCC1)C(=O)N2C.CC1CCC1CN1CCCC1 c1(C(=O)NCCCOCCNC(C(C(CC)CC)C)=O)n[nH]c2nccc(Cl)c12 C=CCC(C)C(=O)NC1(CO)CN(C(c2ccc(SCN3CCCC3)cc2)=O)C1 c1(NC)cncc(CNC(C2CC(C)N2C(c2cccc(CC#N)c2)=O)=O)c1 C12(CNC(C3C(C(=O)OC)C3)=O)CCCC(CN1C(=O)C=Cc1cscn1)C2 C1(NC(C(COC)O)=O)CCCCC1CNC(C1CCCC1)=O c1(OC(c2cn(CCCNC(=O)CC3CCCOC3)nn2)C)ccc(CO)cc1 N1(C(C(COC)C)=O)CCCC1(C)CCC(=O)N(C1CC1)Cc1ccoc1 c1(C(=O)NC(CNC(C(C)OC)=O)CO)cccc(C)c1[N+](=O)[O-] c1(OCC(=O)OCCC=C=C)ccc2c(c1)CCC2 C(=O)(CC1=CCCCC1)NCC(=O)NCC(CC(C)C)NC(C1(CF)CC1(F)F)=O C1(NC(COCCCNC(CN(C(C)C)C)=O)=O)CN(C)CCC1O C1(C(=O)NCCC23CC(CO2)C3)CN(C(c2ccn(CCF)n2)=O)CC1C1CC1 c1(OC)ccc(F)c(C(=O)NC2CC2NC(=O)C(O)CC2CC2)c1F Cc1cccc(C)c1C(O)CNC(C(C1(O)CCCCC1)(C)C)=O CC1(NC(=O)C(=O)NCC(F)F)CN(C(C2CCC2(C)C)=O)C1 N1(C(C(N2CCNC2=O)C)=O)CCC(CF)(NC(c2cncc(CO)c2)=O)C1 Cc1ccc2ncc(C(N3CC(F)(F)CC3CCNC(=O)C(O)C(F)F)=O)n2c1 C(=O)(CC(C)(C)CC(C)=O)N1C2CN(C(C3CCC(OCC)CC3)=O)CC1CC2 c1(C(N2CCC(CN(C(=O)COC3CCOC3)C)C2)=O)cc2n(n1)CCC2 c1(C(C(=O)NC(C2N(C(CCOC(C)=O)=O)CCC2)C)C)ccc(Cl)cc1 C1(C(=O)C(=O)NCCOC(CSCC(=O)OC(C)(C)C)(C)C)CCOCC1(C)C.O c1(C(=O)OC)c(C)nn(CC2CCN(CC(Cc3ccc(OC)cc3)=O)C2)c1C CC1(C)CC(CNC(c2ccon2)=O)CN1C(C1CC2CCC2C1)=O C=CCC(C)(C)CC(=O)N1CCC(=CCNC(c2nnc(C(C)(C)C)s2)=O)CC1 c1(CC)nn(C)c(C(N2CC(NC(=O)CCn3ccnc3C)CC(F)C2)=O)c1Cl C1(C(=O)NC2CC(CC(NCP(C)(C)=O)=O)C2)(CO)CCCCO1 N1(C(CC(C)C)=O)CCOCCC1C(=O)NCC(C)(O)C1CCC1 C(=O)(C1=CC2CCC=CCCC12)NC1CCN(c2nccc(CC#N)n2)C1 N1(C(c2cn(CCC)nc2)=O)CCCC2(CCCN2C(=O)C#CC2CCOC2)C1 c1(C(N2CCN(C(c3c(C(C)C)onc3)=O)CC2)=O)cc2c(F)ccc(Cl)c2[nH]1 Cc1ccc(F)c(CC(=O)NC23CCCC(NC(=O)C(O)C(F)(F)F)(C2)C3)c1 C(=O)(C1=CS(=O)(=O)CCC1)N1CC(CNC(c2ccc(CC)s2)=O)C2C1C2 N1(C(C)C)CCC2(CC1)CC2(C)C(N1CCN(C2CCOCC2)CC1)=O c1(-c2nc(C(C)SCC)nn2-c2ccc(F)cc2)nn(C)cc1[N+](=O)[O-] C=C(F)C1(CC(=O)NC23CC(NC(=O)C(c4ccnn4C)C)(C2)C3)CCC1 c1(C(=O)NCc2cn(CC(N3CC(C(C)O)C3)=O)nn2)ccncc1F C1(=O)C(F)CN1.N1(CC)CCC1C(=O)N(CCCNC=O)CCO.C(C)(C)(C)O Cc1[nH]c(=NCc2cccc(O)n2)sc1C(=O)Nc1cccc(Br)n1 Cc1nscc1CNC(=O)NC(c1ccoc1)C N1(C(COCCOC)=O)CCC(F)CC1C(N1CCSCC1C)=O C1(CC)CCCN(C(c2cnc(C)nc2C)=O)C1C(=O)NCCC[Si](C)(C)C C1(C(=O)O)CC(NC(=O)NC2CSCCSC2)CCO1 CCCC(CC)C(=O)N(C(C)CN(C)C(c1cc(=O)n(C)cn1)=O)C c1(C(=O)OC)ccc(CNC2CC2c2ccccc2Br)c(F)c1 c1(C(N(C2CCCN(C(=O)CC3CCC(=O)O3)C2)CC)=O)ccc(S(N)(=O)=O)s1 C1(NC(C(F)=C(C)C)=O)C(CNC(=O)COc2ccccc2Cl)CCC12CCC2 N1(C(c2cc(F)cc(OC)c2N)=O)CC2CCC1C(NC(C1CC1F)=O)C2 c1(C(=O)NCC2N(C(c3c(C)snc3)=O)CC(F)(F)C2)c(C)sc2ccccc12 Fc1ccc(CCCNC(c2nnnn2C2CC2)CCc2ncccn2)cc1Cl C(c1ccc2occc2c1)=CC(=O)NCC(CNC(C=C(C)C1CC1)=O)(C)O Cc1cccc(C(=O)NCC(CC2CCCC2)C(=O)NCc2ncccn2)c1N c1(OC)cc(C(=O)NC2CC2C(=O)NCc2c(F)cccc2Cl)c(OC)cc1Cl c1(C(N2CC(O)(CCNC(CCOCC(C)C)=O)C2)=O)cn(C)c2ccccc12 c1(Nc2c(CC(=O)NCCC(=O)OC)cccc2)c(C)nn(C)c1Cl C1(CC)CN(C(c2cnc(O)cc2C)=O)CCC1NC(=O)CCc1ccco1 C(=O)(CCCN=C(NCc1ccccc1)NCc1ccccc1)NC Cc1cc(C#N)nc(N2CC(c3ccccc3)(CNC(c3cc[nH]n3)=O)C2)n1 CC(Cc1cnc[nH]1)C(=O)NCC(C1CCOC1)NC(c1ccn(C)n1)=O C(=O)(C(C)O)NCCSCC(=O)NCC(c1cccs1)C c1(C(=O)OCC)ccc(N2CCN(C(=O)CN3CCC(C)CC3)CC2)nc1C Cc1[nH]c(=N)sc1C(N1CC=CC(NC(=O)C=CCOC2CCOCC2)C1)=O CC1CC(C(N2CC(NC(C3(CC4CCC4)CC3)=O)C(O)C2)=O)CCO1 Cc1c(Br)c[nH]c(=NCC(c2ccccc2)c2ccccc2)c1C c1(C(C(=O)NCC)N(c2ccccc2C)CC(C)CC)cccc(C(C)(C)C)c1 C1(C(=O)O)=CC(c2sc(CN3CC4CC(O)CC3C4)cc2Br)=C1 C1(C2CCCCC2)(C(N(C(CCNC(C(C(C)C)OC)=O)C)C)=O)CC1 N#Cc1cc(C(N2CC34CCCC3(CNC4)C2)=O)c2ccccc2c1 N1(C(C(C)(C2CC2)OC)=O)CCC2(CCC2)C(CNC(=O)CCCF)C1 c1(C(=O)OC)c(C(N2CC(n3cc(CNC(=O)CSC)nn3)C2)=O)n[nH]c1C C1(NC(c2c(C)cc[nH]2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC1C C1(CC(=O)N(Cc2cccc(NC(c3coc(Cl)c3)=O)c2)CC)CCC(=O)NC1=O c1(OC)ccnc(OC)c1C(=O)NC1CC2(C1)CN(C(=O)CC(C)(C)C1CC1)C2 CCC(C#N)(CC)C(=O)N1CC(NC(=O)C(C)Cc2cnc[nH]2)C(O)C1 CCC(C)CC(=O)C(=O)NCCN(C(c1sc(C)cc1Cl)=O)C1CC1 c1(C(=O)NC(C)(CNC(C2CCC(=O)N2)=O)CO)cccc2c(O)nncc12 c1(CCC(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2O)nc2ccccc2[nH]1 c1(C(N2CC(C(C(=O)NC(C(O)CO)C3CC3)OC)C2)=O)csc(=NC)[nH]1 C(=O)(C(F)n1ccnc1)NCC(=O)NCC(c1ncc[nH]1)O N#Cc1ccc(C(=O)NCc2ccc(C(=O)NC3CC4CCC3O4)cc2)o1 C1(C(c2n(CC)nnn2)NCC2CC(SC)C2)C(C)(C)C1(C)C c1(C(CNC(CCSCCCC)=O)NC(=O)CC(C)O)cccc(Cl)c1 C1(CNC(c2cncc(N(C)C)n2)=O)CC2CN(C(=O)CCF)CC12 CCC(C)C(CC(=O)NC1CCCC(O)CC1)NC(c1cc(OC)n(C)n1)=O c1(C(N(C(C)CNC(C2CCC(C(N)=O)O2)=O)CC)=O)ccc([N+](=O)[O-])s1 c1(C(=O)NC2C(C)CCN(C(=O)CCCN=[N+]=[N-])C2)cnn2ccc(Cl)c(F)c12 N1(C(C(CC2CC2)NC(C(n2c(C)ccn2)C)=O)=O)CC2(C1)NC(=O)NC2=O Cn1nc(C(=O)NC2COCCC2NC(=O)Cn2cnnc2)cc1C(F)(F)F C=CCCC(C)(C)C(=O)NCCC1CN(C(=O)CC2CCN(OC)CC2)CCO1 C1(C(C)C)CN(C(c2ccc(Br)cc2)=O)CCN1C(C12CC(C(=O)N(C)C)(C1)C2)=O C1(C(N(C2CC(C)(C)C2)C)=O)CC2(CC2)CN1C(=O)Cn1cccc1 Cc1nc(C2CCCC2)sc1C(=O)NCC1CC(NC(C2CN(S(C)(=O)=O)C2)=O)C1 CCCCCCC(CNC(c1ncoc1C)c1nnnn1C)CC c1(C(=O)NCC(C)N(C(c2sc(CC)c(C)c2)=O)C)cc2c(Cl)cccn2n1 N1(C(CCCC(=C)C)=O)CCC2(CC1)CC2CNC(=O)CCc1nncs1 c1(C(N2CCC(C)CC2CNC(C2CC2C#N)=O)=O)cc2c(nc1N)CCCC2 c1(C(N(CC(CNC(C(COC)(C)C)=O)C)C)=O)cc(OC)ccc1F c1(C(N2CC(NC(COC)=O)C(CO)C2)=O)ccc2nncn2c1 c1(CC=C(C)C)cc(C(=O)NC2CCN(C(C3(C)CC3C)=O)CC2O)ccc1F C1(C)(NC(C(CCC)N(C)C)=O)CCN(c2nc(OC)ncc2Br)CC1 CC(C)C(CNC(c1occ2c1CCOC2)=O)N=c1[nH]nc(C#N)s1 C1(C(N(C2CCCC(O)C2)C)=O)CC(C)(C)CCN1C(C1CCNC(=O)C1)=O N1(C(=O)NC2CC(SCC(C)C#N)C2)CCC(c2ccc(F)cc2)CC1 C(C(CC(F)(F)F)NC(c1cncn1C1CC1)=O)NC(CCCOCCC)=O O=C1CN(C(=O)CC2CCN(C(=O)C=CCN3CCOCC3)C2)CCN1CCO c1(C(=O)NCC2N(C(C3N(C(C)C)C(=O)CC3)=O)CC2)cccc(C#N)n1 c1(C(=O)NCCCCC(=O)NC(CC=C)(C)C)c[n+]([O-])c(C)cn1 c1(-c2nc(C(c3cc(Cl)ccc3Cl)NC)on2)ccc2c(c1)C(=O)NCCO2 c1(C(=O)NC(C(=O)NC(c2n(C)cnn2)CO)C2(C)CC2)cc(Cl)cn1C c1(C(=O)OC)cnc(Cl)cc1NC(C1CCCN1C(c1scnc1C)=O)=O C1(C(=O)NCCN(C)C(C2CC(=O)N(C3CCCC3)C2)=O)CCC2(CCC2)CO1 C(=O)(C(C(C)O)NC(C1CCCN1C(C)C)=O)NC1CCN(CCC)C1 Cc1cn2c(n1)C(C)CC(C(=O)NC1CN(C(C3(N(C)C)CCC3)=O)CC1O)C2 c1(C(=O)NCC2C(CNC(=O)CN3CCC(O)CC3)C2)ccc(F)c(Cl)c1F C(=O)(CCC(=O)NN(C)C)N1CC(CNC(C2(C(C)C)CCCC2)=O)C(C)CC1 Cc1nc(C)c(C(=O)NC(c2nc(C(C)(C)C)n[nH]2)C)c(C)n1 c1(C(=O)NCC(C2CCCC2)NC(c2c(CC)occ2)=O)ccn2ccnc2c1 C1(NC(=O)Cc2cscn2)CCCC(NC(c2ccc(-c3ccsc3)nc2)=O)C1 N1(C(CC2CCCN(C(c3cc(C)nn3C(C)(C)C)=O)C2)=O)CCN(C)C(O)C1 C12(NC(=O)CSC(F)F)COCCC1CN(C(=O)CCOc1cccnc1)C2 Cc1c(C(=O)NCCC(O)CNC(=O)CC2CCCOC2)sc2[nH]cnc(=O)c12 N1(C(C2C(C(C)(F)F)C2)=O)CCN(C(C2CCCOC2)=O)C(C(N)=O)C1 C12(C(=O)NC(CCNC(C3CC(C)C3)=O)C)CCCC(C1)OC2 CC(CC(=O)N1CC2C(C1)N2C(c1csc2ccc(Cl)cc12)=O)CC(C)(C)C C(C(CO)(CO)NC(=O)CN(C)C)N(C(=O)C(C)SC(F)(F)F)C.C1(=O)C(C)N1 c1(CCC)cnnc(C(N2CC(CC(C)(C)CNC(C3CC(SC)C3)=O)C2)=O)c1 c1(C(N(C(C)C)CCNC(=O)C(c2ccccc2)F)=O)cncc(C(F)F)c1 O=C(C#CC1CCCC1)N1CC(O)CC1C(=O)Nn1cnnc1 C(CCCC(=O)N(CCOC)CCOC)OC.C(CCCC(=O)NCCO)OC CC(C)(C)C(=O)NC1CC1C(=O)NCC1COC(=O)N1 c1(C(N2CCC(N(C(=O)C(F)C(C)C)CC)CC2)=O)cncc(Cl)c1C C(C(=O)N1CCC(C)C1CNC(c1cc(C(N)=O)c[nH]1)=O)(C(C)C)NC(=O)OC Cc1noc(C(=O)NC(CNC(c2cc(Br)sc2C)=O)C2CC2)c1C C1(NC(=O)OC(C)(C)C)CCN(Cc2cccc(CO)c2)CC1CC#N C(C1=NOC2CN(C(c3nocc3C(C)(C)C)=O)CC12)NC(COCCC=C)=O C(=O)(C(C)(C#N)CC)N1CCC(C(C(=O)NCC(C2CCC2)OCC)C)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(C(=O)NCc2cn[nH]c2)C(C)(C)C1 c1(C(=O)NC(C(C)(C)NC(CC(C)n2ccnc2)=O)C)ccc(=O)n(C)n1 C(=O)(CCCC(C)=O)NCC1(C(=O)NCCSC)CC(=C)C1 N1(C(C(c2cccc(C(F)(F)F)c2)(C)O)=O)CCCNC(=O)C1 C(C(=O)N(CC(=O)N(c1ccc(F)cc1)CC1CC1)CCC)(C(C)C)NC(C)=O c1(CCC(=O)NCC(C)N(C(=O)C(N2CCOC2=O)C)C)c(C)noc1C c1(C(=O)NCC(C)(C2CC2)NC(C(C)n2cccn2)=O)ccc(C#N)[nH]1 C1(NC(C2C(C)(CC)C2)=O)CC2(CCN(C(=O)CC3=CCCC3)CC2)C1 C1(CC(=O)N(CCCC(C)C)C)CCCOCC1 N1(C(c2ccc(SC)cc2)=O)CCOC2CN(Cc3c(O)cccc3Br)CC12 N1(C(CC2N(C(CCC(CC)OC)=O)CCCC2)=O)CCCNC(=O)C1C N1(C(C(C(C)C)CO)=O)CCC(C)N(C(c2ccc(-c3cnn(C)c3)o2)=O)CC1 Cc1cc(C(N2CCCC(NC(C3CC3c3ccccc3)=O)C2)=O)c(Br)s1 N1(C(c2c(C)cco2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2(CC2)C1 N1(C(Cc2ncc(C)nc2)=O)CC2CCN(C(c3cc(Cl)c(Br)cc3Cl)=O)CC2C1 c1(CC)cc(C(N2CCC(CNC(=O)C(C3CCCC3)OC)C2)=O)n(C)n1 CC(C)CC(C(=O)NCC1(F)CC(NC(c2ncoc2Br)=O)C1)C(C)C C1(COC)(NC(C2CCC2(F)F)=O)CCN(C(c2cnn(CCF)c2)=O)C1 N1(C(CC(C)OC)=O)CCC2(CC1)C(NC(=O)CC1(CO)CC1)CS(=O)(=O)N2C N1(N2CCC(N(C(C)=O)CC)CC2)CCCC2(CC1)CC2.c1(CC)cnccc1C=O c1(C(N(CCC(C(C)C)NC(=O)CCC(C)(C)C)C)=O)cnc(N)c([N+](=O)[O-])c1 CCC(CC(=O)NCCC1CN(C(c2nc[nH]c3ncnc2-3)=O)C1)CC(C)C C1(CCCCNC(Cc2c(C)ocn2)=O)CCCN(C(=O)CC(C)N(C)C)C1 C(S(=O)(=O)CCCC(=O)NC1CCOC(C)(C)C1)c1ccc(C)cc1C C1(NC(c2scnc2Br)=O)CCCN(C(C2C3(CC3)C23CC3)=O)CC1 N1(C(C2N(C)CCCC2)=O)CC2(CCC2NC(=O)CN2C(=O)CNC2=O)C1 C1(CC(=O)NC2CC(NC(c3c(C)nn(CC)c3C)=O)C2)CCOCC1(C)C C(N=c1cc(-c2cccc([N+](=O)[O-])c2)nc[nH]1)c1nn(CC)nc1Br N1(C(C(CC)n2cccn2)=O)CCOCC(NC(C2CC(C)(F)C2)=O)C1 c1(C(=O)NC2CN(Cc3cnccc3Cl)CC2O)n[nH]cc1[N+](=O)[O-] C(CC(=O)NCCCn1cc(C)cn1)(CC(C)C)NC(C(C)OCC=C)=O c1(C(N2C(C(=O)NC(c3ccc(F)cc3F)CO)CC2)=O)c(Cl)cc(Br)cc1Cl C1(CC(C)NC(c2cc[nH]n2)=O)CCN(C(c2cncc(F)n2)=O)CC1 C(=O)(C1=CCN(C(=O)CC2CC2(C)C)CC1)NC(CCOC)C N1(C(Cn2ccc(C)n2)=O)CCCN(C(=O)CCc2cccnc2F)CC1C C1(C(=O)O)CCN(Cc2cncc(F)c2Br)C(C2CC2)C1 C(=O)(C1CCCc2nncn21)N(C1C(N(C(COC)=O)C)CCCC1)C c1(C(=O)NC2CCCN(C(CCCOCCC)=O)C2)ccc(O)c(CO)c1 c1(C(N2CCCC(NC(C3C(C)CC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Br c1(C(=O)NCC2(CN(C)C(C3(NC(N)=O)CC3)=O)CC2)ccc2n[nH]cc2n1 N1(C(C23OCC(C)(C2)C3)=O)CCCC(F)(CNC(c2cscc2F)=O)C1 c1(C(N2CCN(C(CC3CN(C)C3)=O)C(CF)C2)=O)ccc(N)c(Cl)c1O C(=O)(CCCC(C)(F)F)N1CCC(NC(c2c(NCC)ccc(Cl)c2)=O)C1 CON(CCO)C(=O)C1CCC(NC(=O)C2=C(C)CC2)C1 C(=O)(C1CCCc2cncn21)N1CC2CCC(NC(C(Br)=C(C)C)=O)CC2C1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(=O)Cn4ccnn4)CC3O)cc12 Cc1ccc(S(=O)(=O)NC(c2ccccc2-c2ccc(C)o2)=O)cc1C C1(C#CC(=O)NCC2(C)CCN(C(=O)C(C)S(N)(=O)=O)CC2)(CC)CC1 C=CCC(C(=O)N1CCCCC(N(C)C(c2nn(C)c3c2CCC3)=O)C1)C(C)C C1(C(C)C)CN(C(C2CCC(N(C)C)CC2)=O)CCN1C(=O)C(=O)N(C)C C1(NC(=O)CCCOCCOC(F)F)CC2(CCCN(C(=O)CC3CC=CC3)C2)C1 C(=O)(C(CNC(C1CC(F)(CF)C1)=O)C(C)(C)C)NCc1n(C)cnc1 c1(C(N2CCN(C(=O)C=CBr)CC3(C2)CC3)=O)ccc2ncccc2c1 N1(C(CC2CC(=O)OC2)=O)CC2CCCN(C(=O)CCC3CCCCO3)C2C1 CC1CCC(NC(c2ccc(C(F)F)o2)=O)CN1C(c1ncc(Cl)nc1Cl)=O c1(CC)c(C(=O)NC2CC(NC(c3cnccn3)=O)C2)cnn1-c1nccs1 Cc1c(CC(N2CCC(CC(=O)N(C3CC4(CC4)C3)C)C2)=O)ncn1C c1(C(=O)NCC2(O)CC(C(=O)NCC(C)C(C)(C)C)C2)ccn2cncc2c1 CCCCCCC(CC)NC(C1(C)CCCN(C(C2CCCSC2)=O)C1)=O CCC(CC(=O)NC1CC2(C1)CC2NC(c1coc(Cl)n1)=O)c1ccccc1 C1(CNC(c2c(C)ccc(C)c2)=O)CN(C(C2COCCOC2)=O)CCC1(F)F c1(C(=O)NCC2(NC(c3cc(C(F)(F)F)cc(F)c3)=O)CC2)cc2cccn2cn1 Cc1cc(C(=O)NCCC(C)N(C(=O)C(n2ccc(C3CC3)n2)C)C)ccc1Cl C1(CC(=O)OCC)Cc2ccccc2N1C(=O)CNC(=O)C(C)CC C(=O)(CC(C)C(F)(F)C(F)(F)F)N1C(CNC(CCSC)=O)CC1 C(C)(N(C)N1CCC2(CCC(O)CC2)C1)c1cccc(OC)c1 CN1CCOCC1C(=O)NCC1(C)N(C(=O)CSC(F)F)CCC1 C1(NC(Cc2ccc(C)s2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 CC1CCCCC1(C)C(=O)NCCn1ccc(C(=O)N(C2CC3CCC2O3)C)c1 C1(CN(C(C2C(C)(CC)C2)=O)C2CC2)CCCCN1C(=O)CNS(=O)(=O)NC Cc1ccc(C(N2CC(NC(=O)Cc3sc(O)nc3O)C(C)C2)=O)c(O)n1 N1(C(C2CSCCS2)=O)CCN(C(c2cncs2)=O)C(c2cccc(Cl)c2)C1 Cc1ccnc2nc(C(N3CCCC(NC(=O)CCOCC4CC4)C3)=O)nn12 C(C(C)(F)C(C)(C)F)(c1n(CCNC(N2CCCCCC2OC)=O)nnn1)OC N1(C(C)CNC(c2ccoc2Cl)=O)CCN(C(=O)CCC2CCOC2)CC1 c1(C(N2CCC(CCNC(c3c(C)cc(SC)o3)=O)C2)=O)ncc(C)cc1C C(=O)(C(CNC(c1cccnc1C)=O)CC1CC1)NC(CCCC)C1CC1 CC1CCC(CNC(=O)CSc2cccc[n+]2[O-])N(C(=O)C=CC2CCCC2)C1 C1(C(N2CCCC(C(CNC(c3ccn(C)c3)=O)(C)O)C2)=O)CC12CCOCC2 c1(OC)cc(OC)nc(N2CCCC(C(=O)Nc3ccc(O)nc3)C2)n1 CCCC(CCC)C(=O)NCC1(CNC(C2CCN(C3CCSC3)CC2)=O)CC1 C(=O)(C(CC(C)(C)C)NC(=O)C=CCOCCOC)N1CCC(O)(CC)C1 c1(C(N(CCC(C)NC(=O)Cc2cnns2)C)=O)ccc([N+](=O)[O-])cc1F Nc1cc2c(cc1C(N1CC3(CNC(=O)CC4CCCO4)CCC1C3)=O)CCC2 C1(C2CCCC2)(C(=O)NCc2ccc(Cl)c(Cl)c2)CCNC1 N1(C(c2oc(CC)c(C)c2)=O)CC(NC(=O)C(COC)OC)CC12CCC2 CCCCCC(=O)N1CCC(C(=O)NCCn2ccccc2=O)(CC)C1 c1(OC)c(CNC(C)CCc2c[nH]c3ccccc23)ccc(I)c1F c1(C(=O)NC(=O)Nc2ccc(NC(C)=O)cc2)c(C)cnnc1O O1NC(=O)C(=O)OCC1.C1(C(c2ccccc2)C)CC(F)(F)C1 c1(C(CC)C(=O)N(CC(O)CN(C)C(C2CCCC2CC)=O)C)cccc(Cl)c1 C#CCCC(C(=O)NCC1CC2CCC(C1)C2)NC(c1nocc1Cl)=O N1(C(C(CCCCC)F)=O)C2CCCC1CN(C(=O)CC(C)F)C2 c1(CNC(=NCCC)NCC2(C(N)=O)CCOCC2)ccc2ccccc2n1 CS(=O)(=O)c1ccc(NC(N2CC3CCCCCC23)=O)cc1Cl c1(C(N2C(C(=O)NCC3(C(C)(C)OC)CC3)CC2)=O)cnn(C)c(=O)c1 c1(C(COC)NC(=O)NCC(C)(C)CSc2ccc(Cl)cc2)ccccc1OC c1(OC)nc(C(N2CCCC(n3cc(COC4CCC4)nn3)C2)=O)cc(C)n1 Cn1ccc2cc(C(=O)NCCC3CCCN(C(=O)COC(F)F)C3)cnc12 C#CCC(C)(CC)C(=O)NCCC(C)NC(C1CCCC1C(C)C)=O C1(C)(C(=O)NC(C)(C)C)CC12CCN(C(=O)Cc1ccccc1O)CC2 C(=O)(CC(C)(C)C(=O)OC)NC(C=CC(=O)Nc1c(CC)n(CC)nc1)C NC1CCc2n[nH]cc2N(C(C2(c3ncccc3Cl)CCC2)=O)C1 c1(NC(c2sc3n[nH]c(C)c3c2)=O)ccc([N+](=O)[O-])c(OC(C)C)c1 C(=O)(CC1OCCc2ccsc21)NCCCCC(C)NC(C1COCCN1C)=O Cc1cc(C(=O)NC2CC(NC(C3(CO)CCOC3)=O)C2)c(F)cc1Cl Cc1ccc(CC(=O)NC2CCCC2NC(C2(C)COC(=O)OC2)=O)cc1Cl N1(C(CC(C)CN(C)C)=O)CC(C)(CNC(=O)CNC(N2CCCC2)=O)CC1(C)C CCC(C)C(O)CC(=O)NC(CNC(C1(C2(O)CCC2)CC1)=O)C1CC1 C(=O)(CC(C)(C(F)(F)F)N(C)C)NC(CCCC)C(=O)NC.C1(=O)CN1 CC1CCN(C2CC2)CC1C(=O)NCc1nc(COc2ccccc2)cs1 c1(C(N2C3C(NC(C(CC)CC)=O)CC(C3)C2)=O)cc2ccccc2s1 C(=O)(C(C)(O)C(C)C)NC(c1cccc(C)c1)CNC(CCN(C)CC)=O c1(CNC(c2n(C)nnc2)=O)ccc(CNC(C2CC(=C3CCC3)C2)=O)cc1F N1(C(COCCC)=O)CCOCC(CNC(=O)CC2CCC(C)(C)CO2)C1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(C)NC(C1CC1(F)F)=O c1(C(N2CC(OC)C(NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)ccc(N)c(F)n1 C(=O)(CCCn1ccnc1)NC1C(CNC(C2(COC(C)C)CC2)=O)C1 C1(NC(C(C2CCCCC2)NC(C(C2CCOC2)OC)=O)=O)(CO)CCOCC1 CCCC(CNC(=O)C(F)OC)NC(c1c[nH]nc1C1CC1)=O C(=O)(C1=NOC(C)C1C)N1CCC(CC#C)(C(=O)NC2(COC)CC2)C1 N1(C(c2cc(C)sn2)=O)CCCC2(C1)CN(C(c1ccnc(C)c1C)=O)CCO2 c1(OC)cc(C(N2CCOCC2CNC(=O)C(C)O)=O)c(C)cc1[N+](=O)[O-] C1(C(N2CCC3CCC(C2)N3Cc2ccccc2)=O)CCc2nccn2CC1 c1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CCC2)cccc(OC)c1O N1(C(=O)CCc2cscn2)CCC(F)(C(=O)NC2(CO)CCCCC2)CC1 c1(C(=O)NCC2N(C(COC)=O)C3C(C2)COC3)cccc(SC)c1[N+](=O)[O-] CC(C)(C)CC(O)C(=O)NC1(CO)CCN(C(=O)C2=CCCCCC2)CC1 Cc1ccc(C(=O)NCC23CC(NC(C4OCCOC4C)=O)(C2)C3)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)(C)CO1)=O)NCc1cc(C)ns1 C1(CC(=O)NC2(CNC(CC3CC(CC)C3)=O)CCC2)CCC2(CC2)CO1 C=CCCCCCCC(=O)N1CC(OCCNC(c2n[nH]c3c2CSCC3)=O)C1 N1(C(C(CC)N(C)C)=O)CCC(C2CCCN2C(=O)Cc2nc(=N)[nH][nH]2)CC1 C1(C(=O)NC(C)C(c2ccc(Cl)cc2)O)C2CCC1(c1ccc(Br)cc1)C2 O=C(CC1=Cc2ccccc2C1)NC1CCCC(CNC(=O)CSC2CC2)C1 C1(CNC(Cc2scc(C)c2)=O)CN(C(C2CC3COCC3C2)=O)CC(C)(C)O1 n1(C(C)CNC(=O)Cn2cc(CNC(C3CC3(F)F)=O)nn2)cc(CO)nn1 c1(C(N(C2CCN(C(c3cnc[nH]3)=O)C2)CCC)=O)cnc(NC)cn1 C1(COCC)CCCN(C(=O)NCC2CCCN2c2ccccc2)C1 c1(C(N2C3CCC(NC(C(C#N)C4CC4)=O)(C3)C2)=O)cc2ccnc(Cl)c2[nH]1 N1(CCNC(C2CC(C)(C)OCC2)=O)CCN(C(C2CCC2CF)=O)CC12CCC2 O=C1NC(C(=O)NCCc2cccc(OCc3cn(C4CCC4)nn3)c2)CC1F Cc1cc(C(=O)NCC2CN(C(C3(c4ccccc4)CNC(=O)C3)=O)C2)oc1C N1(C(c2cn(CC)nc2)=O)CC(CNC(=O)C(N2CCSCC2)C)C(F)(CO)C1 C1(NC(c2ccc(C#N)cn2)=O)CC2CCC1C(NC(=O)C(=O)NCC(F)F)C2 c1(OC)ccc(CN2CCCC(C(=O)Nc3cnn(C4COC4)c3)C2)cc1F C1(N(C)C)CN(C(C2(C)CCCN2C(=O)Cc2ccccc2O)=O)CC12CC2 C1(C)(C(N2CCC(N(C(CC(n3c(CC)ncc3)C)=O)CC)C2)=O)CC(C)(C)C1 c1(C(=O)NCC(C2N(C(C(C=CC)O)=O)CCC2)(C)C)cnn2ccsc12 Cc1ccc2nc(C)c(C(=O)NC3CS(=O)(=O)CC3NC(=O)COC(C)C)cc2c1 c1(C(N(C(C)(C)C(=O)N(CCO)C2CC2)C)=O)cnc(OC(F)F)nc1 c1(C(=O)NCC(C2CCCC2O)NC(C2C(C)C2)=O)ncoc1C1CC1 c1(OC(C)CNCC(c2ccccc2)C)ccccc1CC(C)O c1(COC)cc(=NCC2CCC(NC(=O)CCCC3CCC3)C2)[nH]cn1 c1(OC)cc(-c2noc(Cc3cccc(F)c3)n2)nc(Br)c1 CCC(CC)C(C(=O)N1CCCOC(CNC(C2(C)CCSCC2)=O)C1)OC C1(C(N(C)CC)=O)CC2CCC1N2C(c1cnc(C)o1)=O CN1CC(C)(C)CC1C(=O)NC1CCCCN(C(C2(C)CCC2)=O)C1 c1(OCC(=O)NC(C)CCCNC(=O)COC2CCCC2)cccc(C#N)c1 C(=O)(C(C(=O)N1CCC(C(=O)N(C2(CC)CC2)C)CC1)C(C)(C)C)OCC N1(C(COCCC)=O)CC2CCC1C1CN(C(c3csc(C)n3)=O)CC21 c1(OC)ccc(C=CC(=O)NCC2CC(NC(c3csc(CO)n3)=O)C2(C)C)nc1 CCCC(C)C(=O)NCC1N(C(c2ccccc2Br)=O)CCSC1 CN1CC(NC(=O)C(C2(C)CC2)NC(c2ccc(=N)[nH]n2)=O)C(=O)N1 c1(C(=O)NCCCCNC(C(CCSC)O)=O)cc2ccccc2nc1C(F)F C1(C(=O)N(CCC(C)NC(C2CC2C(=O)OC)=O)C)(OCC)CCOCC1 C1(NC(c2ccc(C3(C(=O)OC)CC3)cc2)=O)CCCCC(c2ccccc2)C1 CC1CCN(C(C2CCC(=O)NC2)=O)C1CNC(C1(C(=O)NC2CC2)CC1)=O c1(C(=O)NCC(c2ccccc2)CNC(C(CC)C)=O)ccc(N)cc1Cl N1(C(CSCC#C)=O)CCC(NC(=O)CN2CCn3ccnc3C2)CC(O)C1 CC(CCCCCO)NC(=O)C(C1CCC1)NC(=O)CCc1ccccc1 c1(CC)nc(C)c(C(N2CC(CNC(c3c(Cl)cnn3C(C)C)=O)CC2C)=O)s1 Cn1cccc(C(=O)NCC2CCCCN2c2nnc(-c3ccccc3)o2)c1=O CC1C2C(CCN2C(c2csnc2Cl)=O)CN1C(=O)Cc1ccccc1 C1(C(N2CC(C3(NC(C4CSC4)=O)CC3)C2)=O)CCOC2(CCCC2)C1 CC1CN(C)CC(C(N2CCC(NC(c3c(C(F)F)cnn3C)=O)C(O)C2)=O)O1 N1(CC(c2ccccc2)C)CCC(C)(NC(=O)NCCc2cccs2)C1 Cn1cnc2c1CCC(C(N1CC(NC(C3CCCC(=O)N3)=O)C(O)C1)=O)C2 Cc1cc(=NCCCN2CCCC2)[nH]cc1S(=O)(=O)NCC1C(F)(F)C12CCC2 C1(C(N(c2nc(CC)cc(C)n2)CCC)=O)CC12CCc1ccccc12 c1(CNC(=O)CN2CCC(F)(F)C(Nc3ncc(Br)s3)C2)ccccc1[N+](=O)[O-] c1(CC(=O)NCCC(C)N(C(c2c(SC)cccc2)=O)C)cc(F)cc(F)c1 c1(C(C(=O)OCCSC)N(c2ccc(F)cc2)C2CC2)ccc(C)c(Br)c1C c1(-n2c(C3CCCN3C(=O)C)nc(CCCCC)n2)ccc2nccnc2c1 S(=O)(=O)(c1ccc(C(=O)NC(C)CNC(=O)C(=Cc2c[nH]cn2)F)cc1)NCC C(=O)(C1=C(Cl)CCOC1)NC1CC1NC(C(C)(C)Oc1cccc(Cl)c1)=O c1(C(=O)NCC#CCNC(CCc2onc(C)n2)=O)ccc2c(c1)nc(O)n2C Cc1c(C(C(=O)NCCC2(C)CC2)N(C2CC2)Cc2ccccc2)n[nH]c1C1CC1 Cc1ccc(CC(N2CCC(n3cc(CNC(=O)C(O)C4CC4)nn3)CC2)=O)cn1 C12(CNC(CSCC#C)=O)CCC1CCN2C(=O)CCOc1cccc(OC)c1 C(CCC(CO)NC(C1CN(C2CCOC2)C1)=O)NC(Cc1n[nH]c(=N)s1)=O Cc1cc(=O)cc(CNC(c2cn(CC(F)(F)F)cn2)=O)[nH]1 c1(CCNC(CCNC(=O)CO)=O)ocnc1CNC(C1CCC(C(F)F)O1)=O C1(NC(c2c[nH]c3ccccc23)=O)CCC2CN(C(C34CC(C3)C4)=O)CCC2C1 N1(CC(=O)NCCCC)CCC2(CCN(C(c3cccc4ncccc34)=O)C2)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2ccn(C(F)F)n2)=O)C(C(C)C)C1 CC1CCC(CNC(C2CCSCC2)=O)N(C(c2ccc(C(F)F)c(F)c2)=O)C1 c1(C(=O)NC2CC(C(C)NC(Cc3cc(C)[nH]n3)=O)C2)ccccc1Br c1(C(C(=O)NCCCC)N(C(C#C)C)CCCC)cc2c(cc1OC)CCC2 C(CN=c1[nH]nc(C2CC2)o1)(CC(C)C)NC(C1CCN(C(CC)=O)C1)=O C1(NC(c2csc(C)c2N)=O)CN(C(=O)Cc2ncsc2Cl)CC1(C)C c1(OC)nc(Cl)ccc1C(=O)NC(C1(O)CN(C(=O)CC2CCC(=O)N2)C1)C c1(C(N(CC(C)NC(C2(O)CN3CCC2CC3)=O)C)=O)cc2c(O)cccc2[nH]1 c1(NCc2sc(C)c(Br)c2)nc(=NC2COC3(CCC3)C2)[nH]c2c(C)nn(C)c12 c1(C(=O)NCC2CN(C(CC3C(C)(C)C3)=O)CC23CC3)nn(CCF)cc1[N+](=O)[O-] N1(C(C(CC)C2CC2)=O)CCC2C(CCCN2c2cc(SC)nc(SC)n2)C1 c1(C(N(CCN(C)CCF)C)=O)cc(C)cc(Br)c1 N1(C(COC2(C)CC=CC2)=O)CCCC(NC(C2CCC23CCC3)=O)CC1 CC(O)(CNC(=O)CCCCCNC(c1cc[nH]n1)=O)C(F)(F)F Cc1nnc2n1C(C(=O)NCCC1(CNC(c3ccc(F)c(Cl)c3)=O)CC1)CC2 C1(COC)(NC(C2CCOC2)=O)CCCN(C(=O)C=Cc2cnccc2C)C1 C1(NC(=O)CC2(N3CCCC3)CC2)CC2(C(=O)NCC3C4COCC34)COC1C2 C#CC(CNC(=O)CCCCCN(C(=O)Cc1ccccn1)C)CC(C)(C)C CC1(C)CC2(CC(C(N3C(CNC(c4ccnnc4)=O)CC4COCC34)=O)C2)C1 C1(C2=CCCCCC2)(C(N(C)CC2(O)CCN(C(C(CCC)(C)C)=O)C2)=O)CC1 c1(C(=O)NC2C(NC(CC(C)CF)=O)COC2)cc(F)c(Cl)cc1Cl C1(N(C(=O)CC(Cl)Cl)CCOC)CCN(C(=O)C(c2ccc(F)cc2)F)CC1 C1(NC(c2ccncc2O)=O)CC(F)CN(C(c2ccc(OCCO)cc2)=O)C1 N1(C(c2ccon2)=O)CC2C3CCC(C2C1)N(C(=O)CSc1ccccc1F)C3 n1(Cc2cn(C3C(NC(C(C)S(N)(=O)=O)=O)CCC3)nn2)cc2ccccc2n1 N1(c2cccc(S(=O)(=O)NCCN(OC)C)n2)CCc2ccc(C#N)cc2C1 c1(CC(N2C(CNC(C3(C)CCC(=O)N3)=O)CC2)=O)c[nH]c2cnccc12 N1(C(Cn2ccc(C)n2)=O)CCC(C)(C)C1C(=O)NCC1(CN(C)C)CC1 Cc1nc(C)c(CC(N2CCCC(C)(NC(C3CCCC(F)C3)=O)C2)=O)c(O)n1 c1(CNCC2N(C(CC3CCN(C)CC3)=O)CCCC2)cc2c(Br)cccc2s1 C1(C(=O)NCC(CO)OC)C=CCN(C(=O)CSC(F)F)C1 c1(CNC(C2(C)CCCN2Cc2nc(Cl)ccc2F)=O)ccc(F)c(C#N)c1 C(=O)(C1CCSc2ccccc21)NC1CCC(NC(CCC(C)(C)O)=O)CC1 c1(C(=O)NC2CCC(F)(CNC(C(C)NC(C)=O)=O)C2)ccc(Br)c(N)c1 C1(C(=O)NCCC(C)(C)CO)CC(NC(=O)C2=CCOCC2)C12CCC2 Cc1nccc(C(=O)NC2CC2CNC(=O)CCCSc2ccccc2)n1 N1(C(C2C(OC)CN(C(CCCCCC)=O)C2)=O)CCCC(C2(C)CC2)C1 c1(C(N2CCC(N(C)C(C3CC3F)=O)C2)=O)coc2c1CS(=O)(=O)C2 n1(CC)c(C)cc2c1CCCC2NC(c1c(C)oc2ccc(Cl)cc12)=O C1(CC(=O)NCCC(C)NC(C=C(COC)C)=O)Cc2ccccc2C1=O c1(C(N2CCCC(N(C)C(C3CC(=O)CCO3)=O)C2)=O)[nH]cc2c1CCCC2 c1(C(N2CCOCC(NC(C=CC(C)C)=O)C2)=O)nnc(O)c2ccccc12 C(=O)(C1(C)COc2ccccc21)N1CCCC(CCn2cc(C(C)=O)nn2)C1 c1(CC=C)cccc(C(=O)N(CCC(=O)NCC2C3COCC23)CCO)c1 C12(C(=O)NC3CC(NC(c4nocc4Cl)=O)CC3O)CCC(CC1F)C2 CCC(C)CCCCC(=O)NC1CN(C(c2cccc3c2OCCO3)=O)CC1O C1(CC=C)(NC(=O)CC(C)OC)CCN(C(C2C(C)OC(C)C2C)=O)CC1 N1(C(c2c(C)nn(C)c2)=O)CCOC2(CCC(NC(=O)Cn3cncn3)CC2)C1 C(=O)(CC1OCc2ncccc21)NCCC1CCN(C(=O)CCCCC(N)=O)C1 c1(C(N2CC(N(C(C(C)S(C)(=O)=O)=O)C)C(O)C2)=O)coc2c1CCCC2 C1(CC(N2C(C)CC(CCNC(C(CSC)C)=O)C2)=O)CCCCC1(F)F C#Cc1ccc(C(=O)N(C(CNC(=O)CCC2CCCC(O)C2)CC)C)cc1C C12(CNC(C(F)=C(C)C)=O)CCC1CN(C(C1(c3ccno3)CC1)=O)C2 c1(CC)cnc(C(=O)NC(CNC(c2cc(COC)nn2C)=O)C2CCC2)cn1 C1(C(=O)NCCC(C)(C)N(C)C)CN(C(C2CC2Cl)=O)CC12CCC2 CC(C(=O)NC(=O)CN(C)C)(C1CCC1)NC(=O)CC1(CC2CCC(=O)C2)CC1 c1(NC(c2cscn2)C)[nH]c(=NC2CCCC(O)C2)nc2c1cnn2C C12(C)CCC(C(F)(F)F)(CC1)NC2c1nnnn1C.c1(CCC)cccs1.CC C1(C(=O)NC2(C3N(C(C(C)CF)=O)CCC3)CC2)CCS(=O)(=O)C(C)C1 c1(OC)cnc(C(N2CCC23CN(C(c2nc(Br)ccc2C)=O)C3)=O)nc1C C(=O)(C(C)(C)C#N)N(CCCNC(C(C)CN(C)C)=O)Cc1ccccc1 C(CCCN=c1[nH]cnc(C)c1Br)NC(COc1cccc(OC)c1)=O C1(CNC(C=NOC)=O)CC(C)(C)CN1C(=O)CS(N)(=O)=O c1(OC)cc(C(c2nnnn2C)NCCc2ccncc2F)ncc1C O=C(C1CCc2nncn21)NC1CC2(C1)CC(NC(=O)COCC1CCCO1)C2 C1(CNC(C(CC#C)(C)C)=O)COCC2(CCN(C(=O)CC(=O)N(C)C)CC2)O1 CCC1=NOC(CC(=O)NCCN(CC(C)O)C(=O)C=C(C)c2ccco2)C1 C1(C(=O)NCC(CCC)NC(c2cc(C)sc2C)=O)CCc2nc(C)[nH]c2C1 C1(CC(=O)NC(CCNC(c2n(CC)ccc2)=O)(C)C)CCCN(C(C)C)C1 C1(C)(C(=O)NCCOCCNC(C(C)NC(c2ccco2)=O)=O)C(C)(C)C1(C)C C1(CCNC(c2cccc(C3CC3)n2)=O)CCCCN1C(C1CCC=CCC1)=O CC(C)(F)C(C)(F)C(=O)NCC1CC(NC(c2cncc3ccsc23)=O)C1 N(C1CCCc2c1cnn2Cn1cc(CN)nn1)C(c1sc(C)c([N+](=O)[O-])c1)=O CC1COCCCN1C(=O)C(CC(N)=O)NC(=O)Cc1ccon1 C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1CC(OCc2cccc(OC)c2)C1 C=CCC(CNC(=O)CC1CCC1)NC(=O)CCCSc1n[nH]c(O)n1 N1(C(C2(COC)CC=CC2)=O)CC(N(C)C(C2CCCO2)=O)C(C)(C)C1 c1(C(N2C(C)CN(C(C3(C)CC3Br)=O)CC2)=O)ccc2ncsc2c1 c1(C(c2n(CC(=C)C)nnn2)NCCCNS(=O)(=O)C2CC2)cccc(OC)n1 N1(C(c2cn(C(C)C)nn2)=O)CCOCC(NC(C2(CCF)CCC2)=O)C1 S(=O)(=O)(c1csc(C(=O)NC(C(C)NC(C23CC(F)(C2)C3)=O)C(C)C)c1)NC N1(C(C2C(C)CCC2)=O)CCCC(C)(C)C1CNC(C1CCCSS1)=O C1(NC(C(=O)NCC)=O)COC2C(NC(C3CNC(=O)N3)=O)COC12 c1(-c2ccc(COc3c(SC)nccc3)s2)cc2cccnc2cn1 c1(C(=O)NC(C)CN(C(=O)CCc2nccs2)C)sccc1S(N)(=O)=O N1(C(C=NOC)=O)CC2CCCC(CNC(c3cc(O)nc(O)n3)=O)(C2)C1 c1(CC)c(C(=O)NCC2CC2NC(=O)NCCCO)cccc1C N1(C(C(COCC)C)=O)CC(OC)CC1C(=O)NCc1c(C)cnn1C C1(C(=O)NCC(N(C(=O)COC2CCCCC2)C)C2CC2)(C(F)F)CCOCC1 Cn1cc(CCNC(c2ccc(Br)cc2)c2nnnn2C2CC2)c2ccccc12 c1(C(C)O)nc(-c2ccnc(N(C)C)c2)n(C2CC2)n1 c1(OC)cc(CC(=O)N(C)CCN(C(=O)C(C)(C)CF)C)cc(F)c1 c1(C(=O)NC(C(=O)N(C)CC2(O)CN(C(CC(C)C)=O)C2)C)ccc(F)cc1F S(=O)(=O)(c1ccc(NC)cc1)N(CC#CC1CCCCO1)C.C1CC1 C(=O)(C(C)C(F)(F)C(F)F)NCC(CC=C)NC(c1nc(SC)ncc1N)=O c1(SC)cc(C(=O)NC2CC(CNC(c3[nH]cnc3C#N)=O)C2(C)C)c(C)o1 C1(C(=O)NC(c2ccco2)C)CC(O)CN1C(C1C=CCC1)=O Cc1nnc(N2CC(c3ocnc3CNC(c3cnc(C)o3)=O)C2)s1 N1(C(COc2cc(C)ncc2)=O)CC2CC1CN2C(c1c(O)cccc1Cl)CCCO c1(CC)cc(C)c(C(N2CCC(NC(C3(c4n[nH]cc4C)CC3)=O)C2C)=O)o1 c1(C(N2C(C)CC(CNC(C(CC#C)CC#C)=O)C2)=O)cnc2cnccc2c1 c1(-c2c(C)noc2)cccc2[nH]cc(CN3CC(c4cc(Cl)cc(Cl)c4F)C3)c12 C1(C)(C(=O)NCCC2C(C)CN(C(c3cccc(=O)o3)=O)C2)CCCNS1(=O)=O N1(C(C2(Cc3ccccc3)CCC2)=O)CCC(NC(C2CC2C2CCC2)=O)CC1 c1(C(=O)NC(C(C(C)C)C)CNC(C2(CF)CCC2)=O)ccc(C#N)cc1F c1(C(=O)NC2CCN(C(C(CC#C)C)=O)CC2)cc(Br)ccc1SCC(C)C C=CC(C)CC(=O)NC(CCNC(=O)C(C)CCOC)C(C)C NS(=O)(=O)C1(C(=O)NCC2(F)CCC(NC(C3CCNC3=O)=O)C2)CCC1 N1(C(C(CC)CC)=O)CC2CN(C(c3cc(C(=O)OC)ccc3Cl)=O)CC2C1 C(=O)(C1=C(Cl)CCOC1)N1CC(CCNC(c2ccc(F)s2)=O)OCC1 C(=O)(C1=CN=C2N=CNN2C1)NCC1N(C(C2=CC(C)(C)C2)=O)CC2(CC2)C1 C1(NC(C(C(CC)C)OC)=O)CC2CN(C(=O)C=Cc3cc[nH]n3)CC2C1 C(=O)(C(C)(C)C(C)O)NC1CCC(CC(N2C(C)(CC)CC2)=O)C1 C(C(CC(=O)NCc1ccc(F)cc1)C1CCC1)NC(CN(C)C1CC1)=O c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)C(C)C)ccc(O)nc1Cl C=CC(CCC)CC(=O)NC(C(=O)NCC1([Si](C)(C)C)CC1)C1CCCC1 C1(C(N2CCC(CCNC(c3cnco3)=O)C2)=O)CC2CCC(C1)S2 c1(C(N2C(C(C)NC(CC)=O)CCC2)=O)cnc2ccncc2c1 CCCC(O)C(=O)N1CCC(CCN(C(=O)CCc2c(C)noc2C)CC)CC1 N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(O)C1 C(CCC(C)C(=O)NC1CC(NC(c2ncoc2C)=O)C1)OC C1(OCC)COCC1N=c1[nH]c(=NCCC(=O)NC2CC2)[nH]c2ccsc12 N1(CC(=O)N(CCC(=O)NCC2(CF)CCC2)C2CC2)C(=O)CNC1=O CN1CCCC(C(=O)NCC2CCN(C(=O)CO)CC2)C1c1ccccc1 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)CC2CCCO2)cn(C)nc1C C1(C(c2n(CCCC(=O)OC)nnn2)NC2CC2)CCC(c2ccccc2)CC1 Nc1ncnc2c1ncn2CCNC(c1ccccc1-c1ccc(F)cc1)=O C(CC1=CCN(C(=O)CN2CCCS2(=O)=O)CC1)NC(=O)CC(C1CC1)C1CC1 c1(CC(CC)NC(=O)C(=O)N(C(C)CS(C)=O)C2CC2)cccc(Br)c1 c1(CC(=O)NC2C(NC(C3C(=C)C3)=O)CC2)coc2cc(C)c(C)cc12 c1(C(=O)NCC23CN(C(C4C(C)C4)=O)C(C2)CO3)cncc2c(O)nccc12 S(=O)(=O)(c1ccc(Cl)nc1)N1C(CC)CN(C(C2CN(C)C2)=O)CC1 C1(C(=O)NCCC(C)NC(C2CCN(CCC)CC2)=O)CCc2n[nH]cc2C1C c1(C(=O)NCCC2(OC)CN(C(=O)CC3CCCC34CC4)C2)cc(Cl)ncc1O N1(C(C(CC=C)C)=O)CCC2C(NC(=O)Cc3ccsn3)C2C1 C1(COC)(NC(=O)CC=Cc2ccc(C)cc2)CCCN(C(C2CCSC2)=O)C1 C1(C(N(CCN(C)C(C2(O)CCCC2)=O)C)=O)C(c2ccccc2)C1(F)F N1(CC(=O)Nc2ccccc2)Cc2ccc(Br)cc2C1 c1(OC(C)C)ccc(C(=O)NCC2CCCN2C(c2ccc[n+]([O-])c2)=O)c(F)c1 n1(CC(=O)NCC2N(C(CCC(=O)NC)=O)CCC(C)C2)c(C)cc(O)cc1=O CC1CCC(F)(C(N2CCC(NC(c3ncccc3Cl)=O)C(CO)C2)=O)CC1 N1(CC(=O)NCC2C(NC(CCc3cc(OC)no3)=O)CCC2)CCCCC1=O N1(C(C2N(C=O)CCOC2)=O)CCN(C(=O)C=Cc2ccc(F)cc2)CC(O)C1 N1(C(c2cc(OC)sc2C)=O)CC(C)N(C(C23CCCCC2C3)=O)C(C)C1 N1(C(COCCC)=O)CCC2(CC1)CCN(C(=O)Cc1cc(F)cc(Cl)c1)C2 Cc1cc(CCC(N2CC=CC(NC(C34CC3COC4(C)C)=O)C2)=O)ccc1Cl Nc1ncc(Br)nc1C(=O)NCC1CCC(NC(=O)CCOCC2CC2)C1 C(=O)(C1CCCn2cnnc21)NCCCOCCNC(=O)CC1(O)CCC1 N1(C(c2cnn(CC)n2)C(=O)NC(C)CC)CCc2oc(C)cc2C1 c1(C(N(C(C)C(C)(C)C)C)=O)cc(CNC(=O)CC(C)C2CCCO2)nn1C C1(C)(CNC(CCC2(CCC#C)CC2)=O)CCCN(C(c2cc(Cl)ncc2F)=O)C1 C1(N(C(C(C)C2CCOC2)=O)C)CCC(C(=O)N(C2CCCC2C#N)C)CC1 c1(OC)nn(C)cc1C(=O)CNC(c1cnn(C)c1F)=O C1(NC)C2CCC1N(C(=O)CO)C2.C(=O)(CCS(C)(=O)=O)OC(C)(C)C.C1(=O)C(CCl)N1 N1(C(CN(C(COC)=O)C)=O)CCC(C)N(C(C2CNC(=O)C(C)(C)C2)=O)CC1 N1(C(C(=O)OCC)=O)C2CN(C(C3CCC(=O)N3C(C)C)=O)CC12 c1(C(=O)NCC(=C2CN(C(=O)COC(F)(F)F)C2)F)cnn2ncccc12 C1(NC(CC2CN(C)C2)=O)CC2CCCC(C1)N2C(c1cnns1)=O C1(NC(C=CCCC)=O)C2CC(NC(C3(C)C=CCC3)=O)CC12 CC(C)CC(C(=O)NCC(O)CCNC(c1ccc(C#N)o1)=O)C(N)=O c1(CN(C)C(c2nnnn2Cc2cccc(Cl)c2)c2cn[nH]c2)ccccc1Br c1(OC)cc(C)c(C(=O)N(C)CC2CCN(C(c3cnoc3C)=O)C2)cn1 C1(CC)CN(C(=O)CC2CCCO2)CC1C(N1CC2(CC2)C1)=O C1(CC(=O)OC2C(C(N(c3cnc(C)s3)C(C)=O)=O)CCC2)CC(=O)NC1=O C(=O)(CC(C(C)C)C(C)C)N1CC(OC)C(NC(=O)CCC2CCN(C)CC2)C1 c1(C(=O)NC2CCCC(NC(=O)COC(F)F)C2)ccc(C(C)(F)F)cn1 Cc1cn(CC(N2CCC(NC(C3CC3c3ccccc3)=O)C2)=O)c(=O)nc1O C1(C2CCN(C(C3CSCCS3)=O)C2)(NC(=O)C(CC(F)F)C2CCC2)CC1 c1(C(=O)NC2CN(C(C)=O)C(C)C2)coc2c(C)cccc12 C1(CNC(c2cc(OC)nc(C(F)F)c2)=O)CC12CCN(C(=O)CC(C)C)CC2 CS(=O)(=O)c1ccc(C(=O)NCC2(F)CC(NC(=O)CCOCC(F)F)C2)[nH]1 O=C(CCCCCO)NCC1(NC(C2(N3CCOCC3)CC2)=O)CCOC1 N1(C(C2(C)CCN(C(C(C(C)C)O)=O)C2)=O)CC2(COC(C)(C)C2)C1 c1(C(N(CC(C)NC(C2CCC2C(F)F)=O)C)=O)c(C(F)(F)F)ncn1O N1(C(CS(=O)(=O)NCC)=O)CCN(C(C2(C#N)CC3CCC2C3)=O)CC(O)C1 CC1=CC(C)CN(C(C2C(C)CN2C(C2CCN(C)C2)=O)=O)C1 Cc1cccnc1C(C)NC(=O)CC1CCCN1C(C1CCC(C(N)=O)C1)=O C=CC1(CC(N2CCOC(CNC(=O)CCOCCOC)C2)=O)CCCCC1 N1(CC(=O)NC(C#C)C)CCN(C(c2cnccc2OC)=O)CC1 C1(NC(CSc2cccc(C)c2)=O)CS(=O)(=O)CC1NC(c1cc(C#N)on1)=O c1(NC(=O)OC)ccc(C)c(C(=O)Nc2ccc(CC(N)=O)cc2)c1 N1(C(c2ccc(CCCCC)o2)=O)CCN(C(C2CC(OC)C2)=O)C(C)C1C N1(C(C=C(CC)CC)=O)CCC2(C1)CN(C(=O)CC1CC3(CC3)C1)CC(C)O2 C1(CC(=O)NC2CCC(CNC(CN(c3ccccc3)C)=O)C2)COC2CC1C2 Cc1ccccc1C(C)(C)C(=O)NCC(C)(C)NC(c1cc(O)n(C)n1)=O c1ccc(NCCC2CCCCO2)cc1.C1(CO)(N)CCC1 c1(C(=O)NCC(C2CC2)NC(C2CC(SC)C2)=O)ccc(C2CCCO2)[nH]1 c1(CC(=O)NC(C)CCCNC(=O)C(C)OCC2CC2)cccc(F)c1O C1(C(=O)NCCC(C)NC(c2cnn3c2OCC3)=O)CC(S(C)(=O)=O)C1 C=CC1(CC(=O)NCCc2cccnc2F)CN(C(C2C(C)C2(F)F)=O)C1 c1(NCCC(=O)NC(CC)C)nc(N2CC(O)CC(C)C2)cc(C)n1 C#Cc1cnc(C(=O)NCC2(C(=O)N(C3CC3(F)F)CC)CC3CCC2C3)c(C)c1 C1(CC(=O)NCCCCC(C)NC(C(C)Cc2cnc[nH]2)=O)CN2CCC1CC2 N1(C(C23N(C(=O)CN4CCC(O)CC4)CC(C2)C3)=O)CC2C3CCC(O3)C2C1 C(=O)(C#CC1CCCCO1)N1CCN(C(c2cnco2)=O)CC1c1ccccn1 c1(SCC(=O)NC2C(NC(CC(C)(C)SC)=O)C2)nc2ccc(C)cc2[nH]1 CC1CCN(C(C2(C)C=CCC2)=O)CCN1C(=O)COCC(C)(C)C N1(C(C(C(C)C)NC(N)=O)=O)CC2(CC2)CC1CNC(C1CC12CCSCC2)=O c1(OCC(N2CC(O)(CNC(=O)C3CC3)C2)=O)cccc(C2CCC23CCC3)c1 CCC(CN(C)C)CC(=O)N(CC(C)CNC(=O)C=Cc1cncs1)C c1(C(=O)NC2C(CC)N(C(=O)Cn3cncn3)CC2)cncc2c[nH]nc12 CN1C(=O)NCC1C(N1CCN(C2CCN(C(c3coc(C#N)c3)=O)C2)CC1)=O C(N=c1[nH]cnc(NC(c2nc(C)c(C)[nH]2)C)c1C)c1c(F)cc(OC)cc1F N1(C(c2c(OC)n[nH]c2)=O)CCC(C)C1CNC(=O)COc1cccnc1 CC(C(C)C(=O)N1CC2(CC(NC(c3cc(C4CC4)[nH]n3)=O)C2)C1)C(C)(C)C c1(CC)cc(C(=O)NCCC2(CNC(=O)C(C3CCCOC3)OC)CC2)no1 C1(C(=O)NCC2CCCC2)CCCN(C(=O)CC2CCS(=O)(=O)C2)CC1 CCCC(C#N)C(=O)NCCCCc1cn(-c2ccc(C)c(Br)c2)nn1 c1(C(=O)NC2CC(NC(C3CN(CP(C)(C)=O)C3)=O)C2)cnc2ncccc2c1 C1(NC(c2c(C)nc(C)s2)=O)CC2CN(C(C3CN(C)CC(C)O3)=O)CC12 c1(NC(N(C(CC)CC)CC)=O)cc2c(s1)CCCCCC2OC C1(C(=O)NC2COCCN(C(c3c(C)nc(C)n3O)=O)C2)CS(=O)(=O)CC12CC2 c1(OC)cccc(CN2CCN(Cc3cc(Cl)ccc3C(F)(F)F)CC2)c1F c1(CC(=O)NCC(C2CC2)NC(C(C2CCCC2)OC)=O)nnc(S)n1C CN1CCc2[nH]nc(C(=O)NCC3(NC(=O)Cn4cccn4)CCOC3)c2C1 CN1Cc2cc(C(N3CCCC3CCCC(F)(F)F)=O)ccc2NC1=O C1(C(=O)NCC2(NC(c3cc(Cl)ccn3)=O)CCCC2)CCS(=O)(=O)C1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C(C3CC3)C2)ccc2sc(C)nc2c1 C(C(C)(C)C(=O)NCC1CCN1C(=O)Cn1cnc(=N)[nH]1)SC Cc1nc(C(=O)Oc2cccc(C(=O)NC(N)=O)c2)sc1C N1(C(C(c2cncnc2)C)=O)CCCC2C(NC(=O)C=Cc3ccco3)C12 N1(C(c2nc(CCC)sc2)=O)CCCC(C2(NC(C3(OC)CCSC3)=O)CC2)C1 N1(C(C2(NC(=O)CCN(CC(C)C(C)C)C)CC2)=O)CCC(CO)C(O)C1.COC O(NC(=O)C(F)C(C)(F)F)C(C(=O)N(C(C(NOC)=O)C)C)CC(C)C c1(N2CC3(CCN(C(Cn4c(C)ncc4)=O)C3)C2)nc(Cl)nc2c1CCOC2 CCC(CC)(CC)C(=O)NCC(C)NC(c1ccc(CN2CCCC2=O)cc1)=O C1(NC(C(CCC)C)=O)CC2CCC(C1)N2C(C)C(=O)NC1CCCCC1 C(N=c1cc(NCc2cnn(C)c2Br)nc[nH]1)C1CC(C)SCC1 Cc1cccc(C(N2CCOC(C(=O)NC(c3ccc(Br)cc3)CO)C2)=O)c1O C1(CCNC(C2C(C)CC(C)O2)=O)CCCN(C(c2nnn(C)n2)=O)CC1 C(=O)(CCCCC(C)(C)OC)NC(CC)CNC(=O)C(COC)NC(C)=O C1(N(C(C(C)=CC2CC2)=O)C)CCCN(C(C2CN(C3COC3)C2)=O)C1 c1(C(=O)NC23CC(NC(C4CC4CCCO)=O)(C2)C3)cc(NC(C)=O)ccc1Cl O=C(CC(F)(F)C(F)(F)F)NC1CCC12CN(C(c1cccc3[nH]ncc13)=O)C2 n1(CCC(N2CCC(N(C)C(c3nocc3Br)=O)C2)=O)ncc2c1CCCC2 C(=O)(CCCCN=[N+]=[N-])N(C)CC1CCCN(C(=O)Cn2cncn2)C1 N1(C(C(CSC)O)=O)CCC(C(O)CNC(C2CC(F)(F)CS2)=O)CC1 Cc1ccc2sc(N3CCC(CNC(=O)C(C)O)C(F)(F)CC3)nc2c1C Cc1nn(C2CCS(=O)(=O)C2)c(C)c1CNC1C(=O)OC2COCC12 c1(COC(C2(C3CCCO3)CC2)=O)csc2cccc(F)c12 C1(CCO)(NC(C(C)N(C)C(c2cscn2)=O)=O)CCNC1 c1(CNC(=O)NC2(CCO)CCCOC2)ccc(Cl)c(F)c1F c1(CNC(=O)NCC2CCC(C(F)(F)F)C2)cccc2ccc(Cl)cc12 C(N=c1[nH]c(N2CCOC(CCF)C2)nc2c1COC2)C1(C)COCCO1 CCCC(CCNC(C1(CC)CCN(C(=O)C(C2CC2)SC)C1)=O)CCC N1(C(c2n(CC)ncc2Cl)=O)CCN(C(=O)Cc2ncoc2C)CC(CO)C1 C(CCC(C)(C)C(=O)NC1CC2(COCCO2)C1)NC(C(C)=NOCC#N)=O C1(O)(C(=O)NCCC(C)CCNC(c2ccc(CO)o2)=O)CN2CCC1CC2 c1(-n2c(C3C(OCC)C3)nc(C(C)O)n2)cc(Cl)ccc1C N1(C(C(C(C)C)OCC)=O)CCC2(C1)CN(C(=O)Cc1ccc(C#N)cc1F)C2 Cc1ccc(F)cc1CN1CCOC(C2CC2)C1.C12CC(C1)C(=O)N2 c1(CC(=O)NCCN(C(=O)CC(C2CC2)C2CC2)CC)sccc1Br c1(Nc2cccc(CNC(=O)Nc3c(C)coc3C)c2)ccc2c(c1)CCCO2 C(=O)(C1CCCc2nn[nH]c21)NCCCCNC(CC(CCCC#C)C)=O CCC(CC)C(C)C(=O)N1CC(O)(CN(C(=O)C(c2ccccc2Cl)C)CC)C1 CC1N(C(C2(CNC(c3ncccc3O)=O)CC2)=O)CCOC1(C)C c1(COC)ccc(C(=O)N(C(CC)C(=O)N2CCC(NC(C)=O)C2)C)o1 c1(C(=O)NCC(O)CCNC(c2ccc(O)nc2Cl)=O)ccc2c[nH]nc2n1 C12(CNC(CCCCCNC(C)=O)=O)CCCC(CN1C(C1COCCO1)=O)C2 CCCCCC(C)NCc1ccccc1-c1nnnn1CSc1ccccc1 c1(C(N(CCN(C(c2ccc(C(=O)OC)[nH]2)=O)C)C(C)C)=O)cc2n(n1)CCCO2 c1(C(=O)NC2CCCC(NCC(N(C)O)=O)C2)cc(-c2nn[nH]n2)ccc1N c1(C(N2CCN(C(CS(CCC)(=O)=O)=O)CC2)=O)cc2cccc(C)c2s1 c1(SC)ncc(C(=O)N(C2CN(C(=O)C(C)C3CCC3)C2)C)n1C c1(SCC(=O)NC(CNC2(OC)CCSC2)C)ccc(C(C)(C)C)cc1 CN1CCc2ccc(C(=O)NC3C4CN(C(=O)Cc5ccc(Br)cc5)CC34)cc21 Cc1cccnc1C(N1C(C(=O)NCC(c2ncc[nH]2)C)CCC1C)=O Cc1ncc(CCC(=O)NC2CCCC(NC(c3cc(CF)on3)=O)C2)c(O)n1 N1(C(=O)CC2COCCO2)CCOC2(CCN(C(C3CCCCO3)=O)CC2)C1 C1(CCNC(CC2C(C)C2(F)F)=O)CCCCN1C(c1cc(C(F)F)no1)=O N1(C(C2=CCCN(C(c3cc(CCC)on3)=O)C2)=O)CCCCCCCCC1 C(=O)(CCOC(=O)OCCCNC(=O)C(C)=CC(C)(C)C)NCC=C C1(NC(C(COC)O)=O)CN(C(=O)C=Cc2cncc(O)c2)C(C)(C)C1 C1(NCCCc2cc(C)no2)CC(C(=O)Nc2ccccc2)C1(C)C C1(NC(C23CC(OC)C(OC2)C3)=O)CC2CCC1CN2C(=O)C(=O)NC1CC1 N1(C(CNC(=O)OCC)=O)CC2CC2C1C(N1CCC(OC)C1)=O C1(NC(=O)NC(CC=C)CC)CCC2CC1C2(C)C C1(C(N(CCCOCCNC(CC2(CC)CCC2)=O)C)=O)CCC(=O)N1 C(=O)(C1=Cc2ccccc2C1)N1CCC(NC(c2ncc(F)cn2)=O)C(CO)C1 CC1C=C(C(=O)NC2CC(CNC(c3ccc(F)cn3)=O)C2)CC1 Cc1ccc(C(=O)NC(C)CNC(=O)C(c2ccccc2Cl)O)c2c1NCCC2 Cc1cc(=NC(=O)C=C2CN(C(=O)CC3CCCCO3)C2)[nH]n1C1CCCC1 C(=O)(C1=NOC2(CCC2)C1)N1C2CC(NC(c3ccc(C)cc3O)=O)CC1CC2 CC1(C)COC(CCC(=O)NC2CC3(C2)CC3NC(c2coc(CO)c2)=O)C1 c1(C(=O)NCC2CCN(C(CSCC#C)=O)CC2)cc(C(=O)OC)ccc1Cl N1(C(c2nc(CNC(C3(CC=C)CCOC3)=O)oc2)=O)CCCC2CC12 C(CCCC)(CC(=O)N(C1CC1)Cc1cccs1)NC(C1C(C)(CC)C1)=O C1(CCC)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN1C(=O)CC(C)O C(C(=O)Nn1cnn(CC)c1=O)N(C(C1CCC2(CC2)C1)=O)CC Cc1nc(Cl)sc1C(N1CCC(CC(=O)NCc2nccnc2Cl)C1)=O C12(CCOC(C3CC(OCCF)C3)=O)CCCCC1C2 c1(-c2nc(CNC(C3(C(=O)OC)CCOCC3)=O)c(C)s2)cc(N)cc(F)c1 N1(C(C(CCC)OC)=O)CC2CC(CNC(C3(N(C)C)CCC3)=O)C2C1 C1(CNC(C(c2cnn(C)c2)OC)=O)CC(F)(CNC(=O)CCC2(C)CC2)C1 CC(CC1CCCCC1)C(=O)NC1(CNC(=O)COc2cccnc2)CCOC1 c1(CC)cccc(C(N2CCC(O)(CN(C)C(C3(OC)CCSC3)=O)C2)=O)c1 c1(C(=O)NC2CCC2CNC(C2CC2F)=O)cccc(N=c2cncc[nH]2)c1 N12C(CCC1(C)C)NC2=O.C(CCNC(=O)OC(C)(C)C)N(C)C c1(C(=O)NC2CCCN(C(CC3CC(=O)NC3=O)=O)CC2)ccn2cncc2c1 n1(CC)ncnc1C(=O)N(CC(C)NC(C1CC1CC(C)(C)C)=O)CC CC1(C)CC(=O)NCC1C(=O)NCC=CCNC(c1ocnc1C1CC1)=O c1(C(N2C(C(C)NC(Cc3nc(CC)sc3)=O)CCC2)=O)cnn(C)c1C c1(CC)noc(CC)c1-c1noc(C(C(=O)NC)SCC)n1.C1C(C)(C)CN1C C1(NC(c2nc(C(C)C)sc2)=O)CC12CCN(C(=O)COCC1CCCCO1)C2 CN(C)S(=O)(=O)NC(c1ccc(F)cc1)(C)C.C1C(=O)N1 C(CC(C)(C)C(=O)NCC1CCC(NC(C2CCCC3CC23)=O)CC1)OC N1(C(C(C2CCCCC2)OC)=O)CCCC(CC(N2CCC(C(C)O)CC2)=O)C1 O=C1Cc2cnc(N3CCC(NC(c4ccnc(Cl)c4)=O)CC3)nc2N1 CCCCCC(O)C(=O)NCC12CCC(CC1)N(C(=O)CC(C)(C)O)C2 c1(C(=O)NCC(C)NC(C(C)C2CCC2)=O)sc(Cl)cc1Br C1(NC(C2(COC)CCCO2)=O)CCCCN1C(=O)C=CCOCCNC(C)=O.C.OC c1(C(=O)NCC2(C)OCCN(C(CN(C)C)=O)C2)cccc2c1CC(=O)N2C c1(C(N2CCC(NC(c3nc(C)oc3)=O)C(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(CCCC)CCCN(Cc2ncoc2C2CC2)C1 Cc1c(C(=O)NC(CO)C(C)NC(c2cc(C3CC3)no2)=O)nn2ccccc12 c1(C(=O)NCC2CCC(C)O2)ccc2c(n1)CCN(C(c1ccc(F)c(F)c1)=O)C2 c1(OC)cncnc1C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)c2ccccn2)C1 C1(CNC(C(CC)OC)=O)CC(C(=O)NCc2nc(C)sc2C)=NO1 C1(CC(=O)NCC2COCC2O)CCN(c2ncccn2)CC1 Cn1cc2c(n1)CC(C(=O)NCC(C(C)(C)C)NC(=O)Cc1ccoc1)CC2 c1(N(C)CC2CCN(C(=O)CC3CCCOCC3)CC2)nc2ncc(Cl)cc2o1 C1(C(F)F)(CNC(C(CC2CCCC2)OC)=O)CCN(C(C2CC=CCC2)=O)C1 C1(CCC(=O)N(CC(CC)NC(=O)C(C)(C)n2ccnn2)C)CC(C)(C)CO1 c1(C(CNC(C(=O)NC(c2ncc(C)s2)C2CC2)=O)C)ccccc1Cl c1(C(=O)NCCSC2(O)CCOC2)ccccc1OC(F)(F)F CC1(CNC2COC(c3ccccc3)C2)CCCCO1 C(=O)(CCC(C)(C)C)N1CCC(CC=C)(NC(C2CC(=O)N(C(C)C)C2)=O)C1 N1(C(c2ncc(OC)nc2)=O)CC=C(C(=O)NCC2(O)CC(O)C2)CC1 c1(C(N(CCCNC(C(CC=CC)C)=O)C)=O)cc2n(n1)CCNS2(=O)=O CCC(C)CC(C(=O)NCCC1(OC)CCC1)NC(c1ncccc1CC)=O C=Cc1ccc(C(=O)NC(CN=[N+]=[N-])C(=O)NCCC2CCCC2(C)C)cc1 CC(CC(=O)NC1CC2CC(NC(=O)CCCN3CCCC3)C2C1)C(C)(C)C C(N=c1[nH]c(=NCC2CCCC2)c2ncccc2[nH]1)C1ON=C(C)C1 N1(C(c2c(C)non2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(F)(F)C(C)(C)O c1(CCC)nc(C(=O)NC2(C)CC(NC(=O)Cc3cnc(C)[nH]3)C2)cs1 CC(F)(F)C(F)(F)CC(=O)NC1CCCC1NC(=O)CCc1nc(=N)[nH][nH]1 c1(CC(N2CC(C)N(Cc3cnn(C)c3)CC2)=O)cc(F)c(Br)cc1F N1(C(=O)CN2CCS(=O)CC2)CCCC(O)(CCNC(=O)C=CC2CCCO2)C1 N1(CC)CCCC1CC(=O)NCCC(C)N(C(=O)CCc1nc(C)cs1)C N1(C(C2(S(C)(=O)=O)CCC2)=O)CCN(C(c2ccc(O)cc2F)=O)CC12CCC2 O=C(CC1OCc2ncccc21)NC1CN(C(=O)CCF)C2(CCC2)C1 C1(NC(c2cc(CNC(C3(O)CCC3)=O)on2)=O)CCCC1C1CC1 c1(OC)cc(N)c(C(=O)NCCN2CCN(C(=O)C=CC3CCC3)CC2)cc1F c1(OC)cc(C(=O)NCCN(CC(C)O)C(=O)Cc2cn(C)nn2)cc(Cl)c1 c1(C2CN(CCc3csc(C(F)(F)F)c3)C2)noc(CNC(C(C)O)=O)n1 C(=O)(CCCCCC#N)NC1CN(C(c2cnc(C)c(N)c2)=O)CC1C c1(NC(=O)NCC(C2CCCCC2)OC)cccc(S(=O)(=O)C(F)F)c1 c1(C(=O)NC2CN(Cc3cnc(Cl)cn3)CC2F)c(I)ccnc1F C(CC)(CCCC(=O)NCc1nn[nH]c1C(C)C)NC(CSCCC)=O c1(C2(C(=O)OCc3ccnc(Br)c3)CC2)c(F)cccc1F C(=O)(CC(C(F)F)NC1(C)CC(NC(=O)OC(C)(C)C)C1)OC C1(NC(Cn2c(C)nnn2)=O)CCN(C(=O)CCN2CCOCC2)CC1O N1(C(c2ccn(CC)n2)=O)CC=C(C(=O)NC(CCO)C2CC2)CC1 Cc1cn(C)cc1C(=O)NCc1cccnc1CNC(=O)CC1COC(=O)C1 CC1CC(NC(=O)CCNC(c2ccoc2)=O)CN1C(=O)C=Cc1cnn(C)c1 C(=O)(C1CCCn2cnnc21)NCC(CO)NC(CCNC(=O)NC)=O C1(NC(C2(SCC)CC2)=O)CN(C(=O)COCc2ccnc(O)c2)CCC1C N1(C(c2c(OC)c(=O)cco2)=O)CCC(F)(F)C(CNC(C2CNC(=O)N2)=O)C1 Cc1nc2c(N3CC4(C3)CN(c3ccc(C#N)nn3)C4)ncnc2[nH]1 C(C)(CO)(C(=O)NCc1coc(C)n1)NC(CC=CC=C)=O C1(C(=O)OC)CCC2(CCC1NCC(C1CC1)NC(=O)OC(C)(C)C)OCCO2 c1(C(=O)NCc2ccc(Cn3cc(Br)cn3)o2)csc(-c2ccncc2)n1 c1(OC)cc(OC2C3CCN(C=O)C32)nc(C(F)(F)F)n1.c1(C(=O)N)cn(C)cn1 C(CN=c1cc[nH]cc1C#N)C1CCN(C(C(C)(C)CC2CCCCC2)=O)C1 C(=O)(CC(C)(C)C)NCC(C)(CC)N(C(C(F)=CCC)=O)CC C1(NC(C(C)CF)=O)CCS(=O)(=O)C12CN(C(c1c3c(c[nH]c1=N)CCC3)=O)C2 C1(SC(C(=O)N(CCCNC(=O)Cn2cnnn2)CC)C)CCS(=O)(=O)C1 N(C(=NCCC(F)(F)F)NCCc1nnc2n1CCOC2)CC(C)C c1(C(N2C(C3CCN(C(c4nc(C)sc4)=O)C3)CCC2)=O)nccc2[nH]ccc12 N1(C(C2N(C)CCC2)=O)CC2CC1CN2C(c1ccoc1C(F)(F)F)=O C=CCCC(C(=O)NC12CC(CCC)(C1)C2)NC(C1CC(C)=NO1)=O CN(C)S(=O)(=O)N(C)CC(N1CCCC(O)(CNC(c2cnccn2)=O)C1)=O c1(OCC)ccc(C(C2C(C)CCN2C(=O)C#CBr)O)cc1 N1(C(c2ccc(C=C)cc2)=O)CCCC2CN(C(c3cccc(=O)n3C)=O)CC12 C1(C(N(C)CC2CCN(C(C3(OC)CC3)=O)C2)=O)CCC(C2CC2)C1 C1(CNC(=O)CC2CC=CC2)CC2COCC2N1C(c1ccc2cc[nH]c2c1)=O C(N1CCCC(CNC(C2CC2c2cncs2)=O)C1)n1ncc(C)c1 N1(S(C(C)=O)(=O)=O)CCC2(C1)CN(S(=O)(=O)c1ccn(C)n1)C2 c1(OC)ccc(CC(=O)N(C(C)CNC(C2(F)CCC2)=O)C)c(Br)c1 N1(C(C(C=C)CC)=O)CCC(NC(c2ccc(C)o2)=O)CC1C1CC1 c1(N2CCCC(OC)C2)ncnc(NCc2cccs2)c1C C(=O)(CCC(C)(F)F)NC(c1cn(Cc2cc(C)nc(C)c2)nn1)CCC C=CCC(C(=O)NC(CNC(=O)C(C1CCCCCC1)O)CC)c1ccccc1 c1(C(=O)NC2(CCNC(C3C(C)C3)=O)CCCC2)cc(-n2ccnn2)ccc1F CCC(CCCC(=O)N1CC=CC(NC(=O)OC(C)(C)C)C1)N(C(=O)CC(C)C)CC c1(C(CCCN2C(=O)NC(C)(C)C2=O)=O)ccc(F)c2c1CNCC2 C1(C(=O)NCCC2CCN(C(C3(CCC)CCC3)=O)C2)CC2COCC(C1)C2 N#Cc1ccc(C(N2CCN(C3CCC3)CC2)C(=O)NCC2CCCO2)c(F)c1 C12(CNC(c3cc(Cl)co3)=O)CCCC1CCN2C(=O)CC(C1CC1)C1CC1 CCCCCCC(F)C(=O)NC1CN(C(=O)Cn2cc(F)ccc2=O)CC1F N1(c2ccc3c(c2)OCCCO3)CCN(C(=NCCC2CCCO2)NC2CC2)CC1 c1(C(=O)OC)ccc(C(N2CC3C(C2)C3(C)C)C(=O)NCCOC2CC2)c(Cl)c1 c1(C(N2CC(CC(C)NC(C(C3CCCC3)OC)=O)C2)=O)nccc(C)c1F N1(C(C2CCN(C)C2)=O)CCOCC(C)(CNC(=O)C(C)(C)c2cccnc2)C1 C(CC(C(=O)NC1(CNC(=O)CCc2cn(C)nc2C)CCOC1)N(C)C)SC N1(C(C(C)OCC(C)C)=O)C2CCC1C(CNC(=O)Cc1ccsc1Cl)C2 O=C(C1=CSCCO1)NC1CCCCC1CNC(=O)COc1ccccc1 Cc1ccc(C)c(ON(C2CCN(C(=O)C=CC3CCOC3)C2)C(CCC)=O)c1 c1(C(N(C(C)CN(C(=O)CCSc2ccc(Cl)cc2)C)C)=O)cccn(C)c1=O c1(NC(c2cc(=N)[nH]c(N)c2)=O)cnn2cnnc2c1 C12(C(=O)NC(C3CCN(C(=O)CCn4cnnn4)CC3)C)CCCC1CC(=O)C2 CN(C)S(=O)(=NCC(=O)NC1(C)CCC(NC(C2CC23CC3)=O)CC1)N=O Cc1ccc(C(=O)NC(=O)CN(C(c2ccc(F)cc2)C)CCO)cc1 C1(C(=O)OC(C)(C)C)CCCN1CCC(=O)NCCC(C)(F)F C12(CC)CN(C(=O)C(C)C)C(CNC(c3coc(C(C)(C)C)n3)=O)(C1)C2 N1(C(c2c(CNC(C(C(C)C)C#N)=O)cco2)=O)CCCNC(=O)C1C(C)C C(C(C)(O)CNC(c1cnn(C2CC2)c1)=O)N(CC(=O)NCC1CCCO1)C c1(OC)cccc(CCC(=O)NCCN(CC(C)O)C(C2CC(F)(F)C2)=O)n1 CN1N=C(CC(=O)N(C)CC2CN(C(c3ccc(F)c(C#N)c3)=O)C2)CC1=O N1(C(C2CC(=C)C2)C(=O)n2c3ccc2cc3)CCCC(C#N)C1.C1(SCC)CC1 C1(NC(CNS(CCOC(C)(C)C)(=O)=O)=O)CCCN(C(c2ccns2)=O)C1 C1(F)(CNC(=O)C=CCn2cncn2)CCCN(C(C2CCS2(=O)=O)=O)C1 C1(C)(C(=O)NC(C)CN(C(=O)CCOCC(F)F)C)CCC(=O)N1 c1(CCC)ccc(C(=O)N(CC(CC)NC(=O)CC2CCCO2)CC)cc1 Cn1nc(O)cc1C(N1CC(CCNC(C2CCC(=O)NC2)=O)C1)=O C1(CC(N2CC(CC(=O)OC)C2)=O)C2CCCC2N1C(C1(O)COC1)=O CC(CN=c1[nH]cnc2c(F)c(F)ccc12)N(C)C(c1ccn(C(F)F)n1)=O C1(CC(=O)NCC2(NC(c3ccc[nH]3)=O)CCC2)CCC(F)(F)CC1 Cc1nc(C)c(C(=O)NCc2nnn(C)c2C(=O)NCC(C)C#N)o1 C(=O)(CCC(=O)COC(c1ccc(CSC(C)(C)C)nc1)=O)OCC N#Cc1cccc(Cl)c1C(=O)OCc1ccnc(O)c1 c1(C(N(CCNC(=O)CCCc2ccc(F)cc2)C2CC2)=O)cc(Cl)ccc1F C(=O)(CCCCCN=[N+]=[N-])NC(C)CN(C(=O)C(C)NC(=O)C(C)(C)C)C N1(Cc2c(N(C)C)ccnc2)CC2CCC1CN2C(c1cc(F)c(F)cc1I)=O C1(C)(c2cccc(OC)c2)CCCN1N(CCO)CC(C)(C)C C1(C(=O)NC(c2ccccc2)C(=O)NC(CCCC)C)CC(F)C(=O)N1 CCC(CC)(CC)C(=O)NCCCNC(c1sc(-c2nc[nH]n2)nc1C(C)C)=O c1(C(N2C(CCCNC(COCC(=O)NC)=O)CCCC2)=O)cc2scnc2[nH]1 Cc1nn(C)c(=O)c(C(N2CCC(NC(=O)CN3C(=O)CCCC3=O)C2)=O)c1C c1(C(N2CCC(O)(CNC(C3(C)CCCC3)=O)CC2)=O)ccc2c(c1)COCO2 n1(C(C)C)cnc(C(N2CCCC2CNC(C2CC2F)=O)=O)n1 c1(C(=O)NCC(C)N(C)C(c2cncc(Cl)c2)=O)cc2c(nn1)CCC2 C(N=c1nc(N2CCC(C#N)C2)c2c([nH]1)CSC2)c1scc(C)c1 C1(C(=O)NC2CC(CNC(c3cc(COC)on3)=O)CC2O)CC12CCOCC2 N1(C(CC(CC)O)=O)CCCC(CNC(c2ccc(-c3ccco3)nc2)=O)CC1 C1(NC(c2ccc(OCCC)cc2)=O)CC2CC(NC(=O)C(C(C)C)SC)C1C2 c1(NC)snc(C)c1C(=O)NC1CCN(C(C2CCCC(OC)C2)=O)C1 C(=O)(CC1CCc2ccccc21)NC(CC(C)NC(c1c(C)cc(F)nc1)=O)C N1(C(c2cccc(SC)c2)=O)CCCN(C(=O)C(C)n2cccn2)CC1C c1(C(=O)OC)ccc(C(N2CCN(C(=O)C=CCF)C3CC23)=O)cc1C C(C)(CCNC(C1(C(=O)C2CC2)CC1)=O)NC(C=C(COC)C)=O N1(C(c2n(CC=C)ccn2)=O)CCC2(CCCN2C(C2CC2(C)CC)=O)CC1 CCC(C)(C#N)C(=O)NC1CC(CC(=O)NCc2ccc(N3CCNC3=O)cc2)C1 c1(C(=O)NC(CC(=O)NC2C(C)(C)C2C#N)(C)C)cc2occc2[nH]1 c1(C(N(CCNC(c2c(C)c(Br)no2)=O)C)=O)c[nH]c2cccnc12 c1(C(=O)NCCC2CCCN2C(=O)Cc2cc[nH]n2)sc(F)cc1Br Cc1ccc(NC(=O)C(C)NCCC2CCCC2(F)F)cc1 N1(C(C(CC)O)=O)CCC2(CCN(C(=O)CCN3CCc4ccccc4C3)C2)C1 C(C)(CN=c1[nH]cnc2ccc(F)cc12)NC(C(CC(C)C)(F)F)=O c1(C(=O)NCC(=CC(=O)N(CCCCCC=C)C)C)cc(C#N)nn1C S(=O)(=O)(c1cc(C(=O)NC(C)(C)C)ccc1F)NC.C12(CCCCC1)C(=O)N2 CC1CCC(C)N1CC(=O)NCC(C)(C1CC1)NC(=O)CN1CCCNC1=O c1(C(N(CCNC(C(CCCOC)C)=O)C2CC2)=O)ccc2occc2n1 Cc1ncc(Cl)cc1CC(=O)N(C1CCCCN(C(=O)CCC(N)=O)C1)C C(CCN=C(NCC(C)Cc1cccs1)N1CCC(C)C(F)(F)C1)SCC C1(O)(CCNC(C(C)CC2CC2)=O)CCCN(C(c2cn(C3CC3)cn2)=O)C1 C1(C)(CNC(CC(C)CF)=O)COCCN(C(c2cnc(N)c(N)c2)=O)C1 C1(CC(=O)NC(C(CC)CC)C)CC(C)(C)CN1C(C12CCC(C1)C2(C)C)=O N1(C(=O)C=CC2CC2)CCC2(C1)c1[nH]cnc1CCN2C(C1CCCOCC1)=O c1(C(C)F)ccc(C(=O)N(C2CN(C(=O)C=Cc3ccncn3)C2)C)cc1 c1(C(N2CCC(C)C2CNC(=O)CCC2CCOC2)=O)ccc2c(c1)C(=O)NC2 c1(C(=O)NCC2N(C(CCN(C)C)=O)CC2)cccc(Cc2nc[nH]n2)c1 C1(CNC(C(CCSC)NC(N)=O)=O)CN(C(=O)Cc2ccsc2)CCC1(F)F O=C(C1=CCCS1)NC12CC1CN(C(C1CCCN1CC(F)(F)F)=O)C2 c1(CC(N2CC(NC(C(N3CCOCC3)C)=O)(CO)C2)=O)noc2ccccc12 C1(C(=O)OC)CCN(S(=O)(=O)NC2CC3(C(=O)OC)C2C3)C1 c1(C(=O)NC2CCN(C(C(C)C#N)=O)C2(C)C)nc2ncc(Br)cn2n1 c1(C(C)C)ccc(C(N2CCC(CCNC(C3(C)CCCO3)=O)CC2)=O)c(O)c1 C#CCCN=C(NCC#CC1CC1)NC(C1CCCO1)C c1(C(=O)NC(C(=O)NCCC(C)N(C)C)c2cccs2)cccc(=O)o1 C1(NC(C=C(C)C)=O)CCC2(CCN(C(c3n[nH]cc3C)=O)C2)C1 C1(C(=O)NCCNC(=O)CC2COCC2O)CCCCC1c1ccccc1 c1(C(=O)OC)cncc(C(=O)Nc2nn(C)cc2OC(C)C)c1.C1CNC(=O)N1.CO c1(C(=O)NC(CC)(C)CC(=O)Nc2ccc(C)c(Cl)c2)ccc(Cl)cc1N N1(C(C(=O)NCC(SC(F)F)C2CC2)=O)CCCCC1CC(F)(F)F c1(C(=O)NCC(CC)(C)NC(C2(N(C)C)CCC2)=O)cc(OC)cc(OC)c1 C(C(CC(C)C)C(=O)NC1CC2(C1)CC2C(=O)N(c1cccc(OC)c1)C)OC CCC(C)C(C(=O)N1CCCC(CCNC(c2sccc2SC)=O)C1)OC C1(c2ccccc2)(C(=O)NC2C(NC(c3cc(F)c[nH]3)=O)C2)CC1(Cl)Cl C#CCCC(C(=O)NOCCCC)NC(=O)C(C)OC(C)=O.C(C=C)O C1(OC)(CNC(C2CN(C)CC(C)O2)=O)CCN(C(c2nc(Cl)cs2)=O)CC1 Cc1ccc(F)c(C(N2CCC3CN(C(C4(C)CCC(=O)CC4)=O)CC23)=O)c1F c1(C(N2CCC(CNC(C(CC)(C)CO)=O)C2)=O)cc(C)c2c(O)n[nH]c2n1 CC1(C)CN(CCC(N2CC(O)(CCNC(C3SCCS3)=O)C2)=O)CCS1 N1(C(C2N3CC(C)N(CC3)C2)=O)CC2(CCCCN2C(C2CCCN2N=O)=O)C1 c1(C(=O)NCCNC(CC2N(C(C)=O)CCC2)=O)cccc2c1CCC2 N1(C(c2cnn(C)n2)=O)CCCC2(C1)CN(C(c1cnc(=N)[nH]c1)=O)CCO2 N1(Cc2cncc(OC)c2)CC2CN(C(c3ccncc3O)=O)C2C1 CC1(C)OC(C(N2CC(NC(c3cnc(O)o3)=O)C3(CCC3)C2)=O)C(C)(C)O1 C(=O)(C(CCCC(C)C)NC(=O)Nc1cccc(N2CCCCCC2)c1)OC C1(O)(C(C(=O)N(CC)CC)(C)C)CCCCC1.C12CCN(C1)C(=O)CSCCO2 CC12CC(C(N3CCC(CCCN4CCOCC4)CC3)=O)(C1)C1(CCC1)O2 C1(C(N(C2CC2)CC)=O)CC12CCN(C(c1sc(F)cc1C)=O)C2 N1(C(c2ncc(OC)cn2)=O)CC(N(C)C(c2cc(Br)c(C)o2)=O)C2(CC2)C1 CCCCC(C(=O)N(CC(Cl)Cl)C)NC(=O)COC1CCCOC1 C(=O)(CCCCCC#N)NCC(C(=O)NCCN1CCC2CC12)N(C)C C1(C2CCCN(C(c3ccc(N)cc3)=O)C2)(NC(C(CC)=CC)=O)CC1 C(=O)(CCCCCC(C)O)N(C1CN(C(CCOC(C)C)=O)C1)C CC1(CNC(=O)C(CNC(C2(C)COC(=O)N2)=O)CC2CCCC2)CCCC1O C1(CNC(CC(c2ccc(C)cc2)C)=O)CC(F)(F)CN1C(=O)C(C)CF N1(C(c2sc3ccn(C)c3c2)=O)CCC2(NC(=O)CCC(C)(C)C)CCCCC12 C1(CNC(C(CCOC)C)=O)(NC(=O)CCC(C)SC)CCC(C)(C)CC1 CC1(C(=O)Nc2ccnn2-c2ccc(F)cc2)CCCN(S(=O)(=O)C2CC2)C1 N1(C(CC2CCN(C(C(=O)NC3CC3)=O)CC2)=O)CCC(O)C(F)(F)C1 c1(N2CCCC(CNC(COCC)=O)C2)nc2ccc(C)cc2s1 N1(C(C(c2cccnc2)C)=O)CCCCC(NC(=O)CC23CC(C2)C3)C1 n1(CC)nc(C(C)C)cc1C(=O)NC(C1CCN(C(c2cn[nH]c2)=O)C1)C CCCCC(C)C(=O)NC1CN(Cc2cnc(Cl)cn2)CC1(C)C N1(C(C23CC(CC)(C2)C3)=O)CC2CN(C(C3(C)C=CCC3)=O)CC2C1 C12(C(=O)NC3C(CNC(=O)CCCCC4CC4)CCCC3)CCCC1OCC2 CCC(CC)C(F)C(=O)NC(C(=O)NCC(F)F)C1CC1 Cc1cc(C(N2CCCC(CO)(Nc3ncnc4sccc34)C2)=O)cc(C)c1F CN1CCCCC(C(=O)NCC(O)CNC(c2cc(C(F)(F)F)ncn2)=O)C1=O C(=O)(C(CCC(C)(C)C)NCC(=O)OC)OCC.C12CC1(C)NC2=O Cc1cc(=NC2CCCN(C(=O)C(F)C3CCCC3)C2)[nH]cc1C#N Cc1nccc(C(=O)NCC(C)NC(c2ncsc2S(N)(=O)=O)=O)c1Cl C1(C(=O)NC2CC(CNC(c3ncccn3)=O)C2)CCn2ncnc2C1 C(CC(C)N=c1cc(C)nc(C2CCC2)[nH]1)NC(c1ccc(OC)cn1)=O CCC(CC)(CCNC(C1CCCC1C(F)(F)F)=O)NC(c1cnnn1C)=O N1(C(C2(COC)CCOCC2)=O)CC(NC(=O)CC2CC(C)=NO2)CC(F)C1 n1(CC=C)cc(C(=O)NC(c2nocc2C(N2CCCC2CC2CC2)=O)C)cn1 c1(CC(=O)NCC2(CCNC(C=C(C)C(C)(C)C)=O)CC2)sc(C)cc1C c1(CC(=O)NCCCCCN(C(CCC2CC(C)C2)=O)C)ccc(Cl)nc1 N1(c2n(C(COCC)C)c(-c3cccc(F)c3)nn2)CC(CO)OCC1(C)C C#CCC(C)C(=O)NC(c1ccccc1F)CNC(=O)Cc1cnccc1CC CN1C(=O)COCC1CNC(=O)NC1CN(C(C2CCCCC2F)=O)C1 Cc1nc(N2CCC(NC(C3NC(=O)CC3C)=O)C2)cc(O)n1 c1(CCC(=O)NCC(CNC(Cc2ccc(C)o2)=O)C)ccc(=N)[nH]c1 C=CCCCCCCC(=O)NCC1CCCCN1C(=O)CC1(c2ccon2)CCC1 N1(C(c2c(C)[nH]c(C)c2C)=O)CCC2(CCC(NC(=O)CC(C)C)C2)C1 C(=O)(C(N)COCCF)NCC(c1ccco1)N(C)Cc1ccccc1 C(C(C(=O)N1CCC(C(=O)NCCC2(SC)CCC2)C1)C(C)(C)C)OCC(=C)C C=CC1CN(C(c2ccnc(C)c2)=O)CC1NC(c1cccc(N)c1C(F)F)=O c1(CC)cc(N2CCC(N(C)C(c3noc(CC)c3C)=O)C2)nc(CC)n1 C1(C(=O)NC(CNC(C(C(=C)Cl)(C)C)=O)CC(F)(F)F)CC2(CO1)CC(F)(F)C2 C1(C(C)C)CN(C(=O)C(O)C(F)(F)F)CCCN1C(c1ns[nH]c1=O)=O C(=O)(C(F)(F)CC)NCC(c1ccccc1)CNC(C12CC(CCOC)(C1)C2)=O c1(C(=O)NC(C)CCCNC(=O)C#CC(=O)N(C)C)n[nH]c2c1CCCC2 C1(C(=O)OC)CCCN(C(=O)C(C)=CCNC(c2cccc(O)n2)=O)C1 c1(C(N(CC(C)NC(c2sccc2C(N)=O)=O)C)=O)cc(Cl)c(N)c(Cl)c1 C(C(C(=O)NC1CC(O)C1OC)NC(c1cnn[nH]1)=O)OC CC1CN(C(C2CCN(C)C2=O)=O)CC(C(=O)N(C2CCCCC2O)C)O1 C(=O)(C1COc2ccc(Cl)cc21)N(C1CCCCC1NC(=O)Cc1csnn1)C Cc1nc(C(=O)NC(c2ccnn2C)C(N2CC(S(C)(=O)=O)C2)=O)ccc1C#N c1(CC)oc2ccccc2c1C=CC(=O)NCCNC(=O)C=C(C)C1CC1 C(C(C)(O)C(=O)N1CCC(CNC(=O)C(c2ccncc2)C)(OC)C1)OC C1(C(C(=O)NCCCC(C)NC(Cc2c(C)scc2)=O)(C)C)CCCN(C)C1 c1(C(=O)NC2C(CC(NOCC(C)O)=O)CCC2)cc(Cl)cnc1O Cc1cccc(OCC(N2CCCC(C(=O)Nc3ccc(Br)nc3)C2)=O)c1 c1(C(N2CCCC(CCC)(NC(=O)CC(C)CF)C2)=O)nccc2occc12 C(=O)(C(C)(C)CCCNC(=O)Cc1ccccc1O)N1CC(C)C(CO)CC1 C(=O)(CCCCCCNC(=O)CCC1CCCN1C)NCCC(C)CO Cc1nn(C2CC2)cc1C(=O)NC1(C(=O)NC(c2ccccc2)C#N)CC1(C)C N1(C(C2ON=C(C)C2)=O)CCN(C(=O)CC2CC3(CC3)C2)CC1CC(C)(C)C N1(C(c2ccc(CC)cc2C)=O)CCC(NC(=O)CC=C(C)C)C(F)(F)CC1 N1(C(C(C(CC)C)O)=O)CCn2c(C(N3CCC4(CCCCO4)C3)=O)cnc2C1 N1(C(C2ON=C(C)C2)=O)CCC(C)(NC(c2ccn(C(F)F)n2)=O)CC1 C(=O)(C1=NOC(c2ccccc2)C1)N(CC(C)(C)NC(c1c(C)nns1)=O)C N1(C(CC(=C)C)=O)CC2(CCCCN(C(C3CC34CC(OCC)C4)=O)C2)C1 Cc1c[nH]c(C(=O)NCC2(CNC(c3c[nH]nc3C(F)F)=O)CCC2)c1 N1(C(c2ccncc2Cl)C(=O)NC)CCN(C2=NCC(C)S2)CC1 Cc1ccc(CCC(=O)N(C)CCN(C(=O)Cc2ccc(Cl)c(F)c2)C)cc1Cl c1(NC2CCC(NC(C(C)C3CCCC3)=O)CC2)ncc2c(n1)CCCC2 C=C1CCC(NC(=O)NCc2cnn(CC(F)(F)F)c2)C1 N1(C(CCN(CCCO)C(c2c(CC)n[nH]c2)=O)=O)CCC(C)C(C)C1 c1(C(=O)NCC=CCNC(C(CC)OC)=O)cnn2c1CCCC2 N1(C(C(C)c2cccs2)=O)CCC(C)(NC(=O)COCc2ccccc2)C1 c1(CN(C(=O)CC2(C)CCN2C(=O)CSC(F)(F)F)C)ncccn1 c1(C(=O)NC2CCN(C(CCN(CCc3cncnc3)CC)=O)C2)scc(C)c1Cl C1(C(=O)Nc2cccc(NC(C3OC4CCC3C4)=O)c2)CN2CCN1CC2 Cc1cn2c(C(=O)NCCC3CN(C(=O)C(C)CC(F)(F)F)CCO3)cnc2s1 C1(NC(c2ccc(-c3cc[nH]n3)s2)=O)CC2C1CCN2C(=O)C=C1CCCCC1 c1(C(=O)NC2CCCCN(C(C=C(COC)C)=O)C2)c(Cl)ccc2ncccc12 Cn1nnc2c1CCC(C(N1CCC(NC(c3cccnc3OC(F)F)=O)C1)=O)C2 CCCCCCNC(=O)C(c1sccc1F)N(C1CC1)CC1CC1 c1(NC(C(C)OC(C(=C)C)=O)=O)ccccc1CCCCC C1(CC(C)Nc2ccn(C3CCCNC3)n2)CCCCN1 C(=O)(C(C)N(C(=O)C(C)OC(=O)CCC1CCC1)CC1CCCC1)OC N1(C(C(C)n2ccnn2)=O)CC(C2CC2)(C(=O)NCC2CCOCC2(C)C)C1 Cc1ccc(C=CC(=O)NC2C3CN(Cc4ncsc4Br)CC23)o1 c1(C(=O)NCCC2N(C(c3ncn(C)c3)=O)CCC2)nn(C)c2ccc(F)cc12 C=CC1(CC(=O)NCCN2C(=O)CCC2=O)CN(C(C2C=CC(COC)C2)=O)C1 N1(C(c2cscn2)=O)CC(F)(CNC(C2(Cl)CC2(F)F)=O)C1 C=CC1(CC(=O)NCC2CCN2C(c2cc(CSC)on2)=O)CCOCC1 C(C(=O)Nc1cc(C)ccc1C)(C(C)(C)C)NC(c1c(CC)[nH]cc1)=O N1(C(c2nc(C)sc2C)=O)CCC(C)(C)C1CC(=O)Nc1ccc(O)c(C)c1 C1(C(=O)NCCC2CCCCO2)CCCC12CCN(CCOc1ccccc1)C2 c1(C2CC(=O)NCC2)ccc(F)c(NCC2CC2(Br)Br)c1 C1(CNC(C(CC)(C)CO)=O)CCC2(CN(C(C3CSC3)=O)C2)O1 C12CCN(CC1C)C2=O.c1(NC(C2(CC)CC(C(=O)OC)C2)=O)cc[nH]c(=N)c1 C1(C(N(C(C(=O)O)C)C)=O)CCC(C(C)C)N1CC.c1(C(=O)NC)c[nH]c(C)c1 CCC(O)C(C)C(=O)NCC(F)CNC(c1cc(C)n(C)c1C)=O c1(C(N2C(CNC(C(COC)O)=O)CC(OC)C2)=O)cc2ncccc2cc1Cl c1(C(C(=O)O)N(C(CC)(C)C)C2CC2)cccc(F)c1F C(C(C(=O)NCCSCCSS(C)(=O)=O)NC(=O)C(O)C=C)SC C12(C(=O)NC3(C)CC(NC(Cc4c(C)noc4Cl)=O)C3)CCC(F)(CC1)C2 C12(C(=O)Nc3cccc(C(=O)NC(COC)(C)C4CC4)n3)CCC(C1)C2(C)C c1(-n2cc(-c3ccc(OC)c(F)c3)nn2)c(F)ccc(Cl)c1N c1(CC)ncc(C(=O)NCc2nc(C(=O)N(C)Cc3nc(=O)o[nH]3)co2)cn1 C(C1CCOCC1)=CC(=O)N(CCC(N1CC(C)(C(=O)OC)C1)=O)C1CC1 C1(CSC)CCN(C(=NCCF)NCC(c2ccc(F)c(F)c2)O)C1 CC1(C(=O)NC(CC(=O)NCCC2(C)CC2(F)F)C2CC2)CC(=O)C1 C1(C(=O)OC)C(CC(=O)NC(C)CN(C)CCC2(C)CCCC2)C1(C)C c1(SC(=O)C(C)C(CC)SCC#C)ccc(-c2nnc(C3CC3)n2N)cc1 N(C(=NCCOC)N1CCC(C2(O)CC2)CC1)CCC1(COC)CCCC1 c1(OC)ccc(F)c(C(N2CCCC(CN(C(=O)C(Br)=C(C)C)C)C2)=O)c1F C(CN=c1ccnc(N(C)C)[nH]1)(c1ccccc1)NC(c1c(C)nns1)C CCCC(C(=O)N1CCCC1CN(C(C1CC=CCO1)=O)C1CC1)NC(N)=O CCCC(C)(C)CC(=O)NCCCOCCN(C)C(C1(CO)CCOC1)=O CN1C(=O)OCC12CCN(C(c1cnn(C3CCC3)c1)C(=O)NC1(C)CC1)C2 C12(NC(c3c(C)nc(O)[nH]3)=O)CCCN(C(C3(CC(C)C)CC3)=O)CC1C2 c1(-c2n(CCOC)cnn2)ccc(-c2noc(CC(C)C)n2)cc1 c1(C(=O)NC2C(NC(c3nc(CC)oc3)=O)CC2)cnc2sc(C)c(C)n2c1=O C1(CNC(c2cnc(CC)[nH]2)=O)CN(C(=O)CCc2cccc(C)c2)CC1C Cc1n[nH]c(C)c1CCC(=O)NC1CCCC(C(=O)NCC2CCC(C)C2)C1 C1(CN(C(c2c(SC)csc2)=O)C)CCCCN1C(=O)C(C1CCCO1)C1CC1 Cc1nc2cc(NC(=O)CC3COCCN3C(c3scnc3C)=O)ccc2o1 C(=O)(CC(C(F)F)n1ccnc1)Nc1nc(C)n(C)c1.C1CCCCN1C N1(C(=O)CC2CC(C(=O)NCC(N3CCCC3)C)C2)CCC(C)(CO)C1 N1(C(C2(NC(CCOCCOC)=O)CCCC2)=O)CC2(CC(CO)CO2)C1 CC1CN(C(=O)C(c2ccccc2)O)CC(C)C1N=c1nc[nH]s1 C1(C(=O)NCC(CN(C(Cn2c(C)ncc2)=O)C)O)CC12CCC1(CC1)CC2 CC(C)CS(=O)(=O)CC(=O)N1CC(O)(CNC(c2csc3ccncc23)=O)C1 Cc1ccc(C)c2c1N(C(=O)NC1CC(O)C(S(C)(=O)=O)C1)CCC2 N1(C(CCNC(COC)=O)=O)CC2CC(NC(=O)CCc3ccncc3)C1C2 C1(CNC(CC(COC)(C)O)=O)CC2(CCC2)CN1C(=O)CCc1cc(C)on1 C(=O)(C(F)(F)Cc1ccc(Cl)cc1)N1CC(C(C)(C)C)C1 N1(C(=O)NC(c2ccc(O)nn2)C)CCC(Cc2ccccc2Cl)CC1 CCCC(CCC)CC(=O)NCC=CCNC(=O)CCc1ncc[nH]1 C(CCC(N)=O)(C(=O)NC(C)(CNC(=O)CCCCCF)C1CCC1)NC(C)=O c1(C(N2CCN(C(C(CCSC)OC)=O)CC2C)=O)cc(F)cc(F)c1O C1(NC(C(C)SCCCC)=O)CC(NC(C2CC=CCO2)=O)C(O)C1 Cc1c(C(N2C(C(=O)NCc3cc(F)ncc3Br)CC3CC23)=O)cncc1Br N1(C(CSC(C)C)=O)CCCC1(C)CNC(=O)CCOCCOCCCO c1(OCC)nc(N2CC(C(C)NC(=O)C(C)(C)c3ccccc3)C2)ncc1Cl N1(C(C2(C)CCOC2)=O)CCCN(CCNC(=O)C(=O)NCC2CC2)CC1 c1(CC)cccc(C(=O)NCC2CN(C(=O)C(=O)NC3CC3)CC2O)c1F N1(C(C(C)=C2CCC2)=O)CCC2CCCC(C1)N2C(=O)CCc1cnn(C)c1 C1(COC(c2cc(C)oc2C)=O)Cn2ccnc2NC1=O c1(N(C(c2[nH]nc(C(F)(F)F)c2C)C(=O)NCCSC)C)cc(C)ncc1C CS(=O)(=O)c1c[nH]c(=NC2CN(C(c3cnc(C(C)(C)C)o3)=O)CC2C)cn1 C(=O)(C1CCc2c(Cl)cccc21)N1CC(NC(C2CC=C(C)CC2)=O)C(C)C1 N1(C(C(CC)(C)OC)=O)CCN(C(c2ccc(C3CC3)s2)=O)CC12CC2 C1(NC(c2ccc(OC)nc2Cl)=O)C2CCC1CN(Cc1ccnn1C)C2 N1(C(C(=O)N(C)C)=O)CCN(C(=O)CC2CCC(=O)O2)CC(O)C1 Cc1ccc(S(N)(=O)=O)cc1C(=O)NC12CC1CN(C(C1(C#N)CC(C)C1)=O)C2 N1(C(C2(OCC)CCC2)=O)CCOCC2(COCCN2C(c2ccco2)=O)C1 c1(C(=O)NCC2CC(NC(CC(=C=C)C)=O)C2)cc(Br)cc2scnc12 CC1(C)C(CC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1O N1(C(C)=O)CS(=O)(=O)CC1C(N1CCC(CNC(C2(C)CC2C)=O)C1(C)C)=O C1(C(=O)NCC#CCNC(CC2(C)CCCO2)=O)OCC2COCCC12 C(CCC(O)C(=O)NOCCN(C)C)NC(c1cnc(OC)s1)=O CC(C)CC(C(=O)N1CCN(C(c2sccc2C#N)=O)CC1C)C(C)C C(=O)(C(C)(O)Cc1ccccc1)NCC1C(NC(c2n(CC)ncc2)=O)C1 CCC(CC)C(C)C(=O)NCC1CN(C(=O)Cc2cc(F)ccc2OC)C1 N1(C(c2c(C)nc(C(C)C)cc2)=O)CC2CN(C(c3cnoc3C)=O)CC2(C)C1 N1(C(C(CC)COC)=O)CCCC(N(C)C(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(C(N2CC(CC#C)OCC2)=O)N(C(c2cc[nH]n2)=O)CC12CCCC2 C1(CC(=O)NCCC(C)NC(c2cn(CCC=C)nn2)=O)CCCC(=O)C1 Cc1cc(C)cc(C=CC(=O)NC2CC2NC(c2cccnc2N)=O)c1 c1(CCN(C(=O)NCC2CC(N)C2)CC2CC2)ccccc1[N+](=O)[O-] C(=O)(C1=C2CCN=C2NC=C1)N1CCC(C(C)NC(c2cncc(C#C)c2)=O)C1 N1(C(=O)OC(C)(C)C)CC2C1COC2=O.c1(C(CN2CCCCC2)O)cccnc1 C1(F)(CNC(C(C)NC(CC)=O)=O)CCC(NC(=O)C=Cc2cccn2C)C1 N1(C(C2(CC)CC2)=O)CCC(C)C(NC(c2cc(C3CCCCC3)[nH]n2)=O)C1 c1(CNCC2N(C(C3CC(=C)C3)=O)CC2)c[nH]c2cccc(OC)c12 CC1(CO)CC(O)CN1C(C1CCC1)=O.O1NC(=O)CNC(=O)C1 CCCC(CC)C(=O)N1CC(CCNC(=O)CNC(C)=O)C(C)C1 C1(CNC(c2c(CC)occ2)=O)CN(C(=O)CSc2n[nH]c(O)n2)CCO1 C1(C(=O)NC2(CNC(c3ccc(CC(C)C)o3)=O)CCC2)CC2(C1)CC21CCC1 CCCCC(CC)CC(=O)NCC=CC(=O)NCCC1(C)CC1(F)F c1(OCC)ccc(Br)cc1C(=O)NC(c1nc(C2CC2)no1)(C)C N1(CC(=O)N(CC#N)Cc2scc(C)c2)CCc2c(Br)cccc2C1 N1(C(CN(CC(C)C)C(C2CC3(CCC3O)C2)=O)=O)CC2(CCC1CO)CC2 c1(CC)ncoc1C(=O)NC(C1CCOC1)CNC(c1cc(Cl)ns1)=O C(=O)(C(O)C(C)(C)CC)NC12CC(CN(C(C3CCCN(C(CC)=O)C3)=O)C1)C2 c1(C(CN)C)cnn(C)c1.C(C(=O)N(CC(C)O)CCSC)=CCOC CCCCC(F)C(=O)NCC1CCCCC1C(=O)NOC1CCCNC1=O CN1CCC2CN(C(=O)CC3(CNC(=O)C=Cc4ccoc4)CC3)CC2C1 Cc1c(C(=O)N(C)CCNC(=O)CCCc2nccs2)cccc1F C1(CC(N2CC(NC(c3cc(OC)n[nH]3)=O)C2)=O)C(=O)N(C)N=C1C CC(CC(F)(F)F)C(=O)NC1CCC(CNC(c2ccc3[nH]ccc3n2)=O)CC1 c1(C(=O)NC2(CCCC(=O)NCc3ncc(C)o3)CCC2)ccnc2cc[nH]c12 Cc1nc(=NC2CCCCC2CNC(c2coc(CCC(F)(F)F)n2)=O)s[nH]1 C#Cc1cccc(CC(=O)NCC2(C)CCCN(C(=O)C(O)CCSC)C2)c1 N1(C(Cc2ccn(C)n2)=O)CCCC12CCCN(C(C1CCC(C)(C)CO1)=O)C2 N1(C(c2nc(C)oc2)=O)CCC(O)CC1C(=O)NC1CCC(C)CC1 C1(C(=O)NCC2(OC)CC2)COCC1NC(C1(CO)CCCO1)=O C1(C)(NC(c2c(C)c[nH]n2)=O)CCN(C(=O)C2=CSCS2)CC1 c1(C(N2CCC(C(C)NC(c3c(CC)sc(=N)[nH]3)=O)C2)=O)cnc2[nH]cnc2c1 N1(C(c2c(C)snc2)=O)CCCC(O)(CNC(c2ccc(CCF)cc2)=O)CC1 C1(C(=O)NCC=C(Cl)Cl)(CNC(C2CCCCS2)=O)CC12CCC2 c1(C(=O)NC(CC)(CNC(C2(C)CCC2)=O)CC)cc(Cl)c2ccncc2n1 c1(C(=O)NCC2(O)CCN(C(C3=CCC(C)CC3)=O)C2)cc2c(F)cccc2s1 Cc1cccnc1C=CC(=O)NC1CCC1NC(=O)CC(C)C1CCCC1 c1(CC)cscc1C(=O)NC1CCCC1CC(=O)NCCC1SCCS1 C1(CC(=O)NC2(COC)CN(C(C3CC(O)CN3C)=O)C2)COCC(C)O1 C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(F)CC2CCOC2)CC1C c1(C(=O)NCC(CO)NC(c2ccc(C)cc2O)=O)cc([N+](=O)[O-])c(C)cc1C C1(n2cc(C3CCN(C(C4(C)CNC(=O)C4)=O)CC3)nn2)CCC(F)(F)CC1 c1(NC(=O)NCCSCc2ccccc2)c[nH]cc1Br C12(NC(C3(CC)CCNC3=O)=O)CCCC(CN(C(c3ccncc3O)=O)C1)C2 c1(C(N2CC(C)C(NC(=O)CN(C)C)C(C)C2)=O)cc2cccc([N+](=O)[O-])c2[nH]1 N1(C(C2C3(CCN(C(c4c(C)ocn4)=O)C3)C2)=O)CC2CC(C(=O)O)C(C2)C1 N1(C(C2(C)CC3CC3C2)=O)CC2(CC(NC(=O)C(C(C)(C)C)NC(N)=O)CO2)C1 Cc1[nH]c(Cl)nc(=NC2CN3CC23)c1C#N.C(=O)CS(=O)(=O)C(C)(C)C N1(C(=O)Cc2cc[nH]n2)CCC2(CC1)CN(C(c1cc(F)cc(Cl)c1O)=O)C2 Cc1cc(OC(c2cccc(Oc3ccccc3)c2)C)nn1C Cc1cc(CNC(=O)C(=O)NC(c2cnn(C)c2)C)c(C)s1 CCC(C)(C)C(O)C(=O)NCC1CC(C(=O)NC2CCn3cncc3C2)=NO1 N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCC(CC)CC2)=O)C1 N1(C(C(=O)N(c2cccnc2)CCOC)=O)CCC(c2ccc(C)s2)C1 C1(C(F)(F)C(=O)NCC=CCNC(C2CC2[N+](=O)[O-])=O)(N(C)C)CCCC1 N1(C(C2(C#C)CCCC2)=O)CC2CC(NC(C3(C)CCN(C)C3)=O)C1C2 C1(CN(C(=O)CC2CC(F)C2)CC)CCN(C(=O)CC2(N(C)C)CCCC2)CC1 C(=O)(C(C(C)C)n1ncc(N)n1)NCC(=C)CCNC(C1C(C)C1C)=O c1(-c2c(OC)c(F)c(F)cc2)n[nH]c2cccc(C(=O)NCC(O)C(F)(F)F)c12 C1(C(=O)NCC(CC)(CC)NC(=O)C(C)N2CC(C)C2)CC2C=CC1C21CC1 C1(CCCNC(c2ncn(CC)c2)=O)CN(C(c2nnsc2SC)=O)CCO1 Cc1ccc(C(N2CCC2CC(=O)NC23CCC(CC2F)C3)=O)c(C)c1 C(=O)(C1COc2ccccc21)N(CC(C)NC(C1CC=C(C)CC1)=O)C N1(C(c2c(N)non2)=O)CCOC(CCNC(C2CC3CC3C2)=O)C1 C(CC(CNC(=O)C(C)(C)NC=O)NC(=O)C(Cc1ccsc1)NC=O)OC c1(C(=O)NCC(CCOC)NC(=O)CCC2CCC2)ccc2c(c1)CCC(=O)N2 C12(NC(CC3(C)CCN(C(C(CC=C)C)=O)C3)=O)CCCC1OCC2 CC1=NOC(C(=O)NC2CC(C(=O)NCc3cnc(C)[nH]3)C2)C1 CC(C)C(Cc1ccccc1)N=c1cc[nH]c(=NCCCCF)[nH]1 N1(C(c2cccc(C)c2O)=O)CCC(C2(NC(=O)CCn3cc(Cl)cn3)CC2)C1 Cc1cc(C(N2CCC(N(C)C(c3ccn(C4CC4)n3)=O)C2)=O)c2c(c1)CCC2 c1(CC)nn(C)c(C(N2CC3CC3(CNC(=O)CN3CSCCSC3)C2)=O)c1Cl CC1CN(C(C2CC(C)(O)C2)=O)CCCN1C(c1ccc(S(C)(=O)=O)[nH]1)=O C(c1cc(Cl)cc(Cl)c1)=CC(=O)N(CCC)CCNC(C1CC(O)(C(F)F)C1)=O CCC(CC(=O)N1CCC(C(=O)N=c2cc(C)n(C)[nH]2)C1CC)C(C)(C)C C12(C(=O)NCCC3CCN(C(C(COC)OC)=O)C3)CC3CC1C2C3(F)F n1(CC)cnc2c(N(C)Cc3nc(C)ns3)nc(N3CCC(C)CC(C)C3)nc12 c1(CN(C(CCC2(NC(C(C)OC(C)=O)=O)CCC2)=O)C2CC2)cnn(C)c1 c1(C(N2CC3C(CNC(C=CSC)=O)(C3)C2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] O(N(C(=O)C1CC(C)(C)CN1C(=O)CC(C)CC1CC1)C(C)C)CC N1(C(C2(CSC)CC2)=O)CC(CNC(C2(C)CC=CC2)=O)C(F)(F)C1 CCCCCCCS(=O)(=O)NC(c1ncc(F)cc1F)C Cc1ccc(SC(C)C(N2CCC(Nc3nccc(CO)n3)C2)=O)cc1 CC1(C)CC=C(C(=O)NC2CC2NC(C2CC3(C2)CC(C)(C)C3)=O)CC1 CCC(C)CC(C(=O)NCc1ccc(SC)o1)NC(C1CCCC(=O)C1)=O c1(CCC(=O)NC(C(C)NC(=O)Cn2ccc(C3CC3)n2)C)ccc(F)cc1F C12(NC(C3CC(C#N)C3)=O)CCCC1CN(C(c1sccc1F)=O)C2 c1(C(N2CSCCSC2)=O)ccccc1-c1cccc(CO)n1 c1(C(=O)NCC2OCCC2C(=O)NCC2C=CCCC2)ccc2n[nH]cc2c1 N1(C(C(C(C)C)O)=O)CCC(n2cccn2)(CNC(c2cc(C#N)no2)=O)CC1 N1(C(c2ccc(C(C)=O)s2)=O)CCOCC1CNC(=O)C(C1CCOCC1)C c1(C(=O)NC(CC)C(OC)OC)cc(S(=O)(=O)N2CCCC2)ccc1F c1(C(N(CCNC(C=CC(=O)OC)=O)C2CC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 c1(CSC)ccccc1C(=O)NCC(O)CNC(c1cc(C2CC2)cs1)=O N1(Cc2cc(C)cc(C)c2)CC2(CN(C(c3coc(C)n3)=O)CCO2)C1 C1(C(N2CCCC(CCNC(C3(C)CC3(F)F)=O)C2)=O)CCCC12CCOCC2 C(CN=C(NCC1(c2ccc(F)cc2Cl)CC1)NC1CCCCC1C)OCC#C c1(CC(=O)N(CC(CC(=O)O)C2CCCCC2)c2scc(C)n2)cccc(C#N)c1 c1(C(=O)NC2(C)CCCCC2C(=O)NC2CCC3(CC3)C2)cccc2[nH]ncc12 O=C(CCS(=O)(=O)c1ccc(F)cc1)N1CCC(C2CC(NC(C3(F)CC3)=O)C2)C1 c1(NCC2(CNC(CC3CCC(C)C3)=O)CCCC2)nnccc1C#N Cc1cc(C(N2CCN(C3CCN(C(=O)CCS(C)=O)C3)CC2)=O)ncn1 C1(NC(C(C)C(F)F)=O)CN(C(c2ccnc(OC3CC3)c2)=O)CC(C)(C)C1 C1(C(N(C)Cc2c(C)nsc2)=O)COCCC1NC(c1nonc1N)=O c1(C(=O)NC23CC(CNC(C4C(C)(C)C4C#N)=O)(C2)C3)n[nH]c2c1CCCCC2 c1(N2Cc3c(CC)cccc3C2)[nH]c(=NCCCCCCCO)nc2scnc12 C1(C(=O)NC2(CC=C)CCCN(C(=O)CCC)C2)CC2(CCCC2)CO1 Cc1sc(-c2ccncc2Cl)nc1CN1CCN(C(=O)Nc2ccccc2)CC1 C1(CCCCCCO)C(=O)Nc2ccc(OC)c(c2)CN1C.C1(CC)CCOCC1 c1(CC(=O)N(C(CN(C(C2N(C(C)=O)CC2)=O)C)C)C)cccnc1 C1(C(N2CC(O)(CN(C(C(CCCC)(C)F)=O)C)C2)=O)CCc2c(cnn2C)C1 c1(C(N(CCNC(C2C(C(=O)OC)CCC2)=O)C2CC2)=O)cn(C)c(=O)cn1 c1(SC)cc(C(=O)NC(C)(CNC(C2CCS(=O)(=O)N2)=O)C2CC2)ccc1F N1(C(c2cnc(C(C)C)s2)=O)CCC(NC(=O)CCCN2CCCCC2)C(O)C1 CC1(C)CCC(NC(=O)NC(C)(C)C(=O)NCc2ccccc2)N(C(N)=O)C1 C1(NC(CCC(=O)NC)=O)CCN(C(c2c(CO)noc2C)=O)C12CC2 C(=O)(CCCCCC(C)(C)C)N1CC2CN(C(c3c(CC)occ3C)=O)C2CC1 CC1CN(C(=O)CSc2ccccc2)CC1NC(=O)Cc1nncn1C Cc1nn2c(c1C(=O)NCCCN(C)C(c1coc(Cl)n1)=O)CCCC2C c1(C(N2CC3C(CNC(C=CC=CC)=O)(C3)C2)=O)ccc(Cl)c(C#N)c1 c1(COC(=O)Cc2ccc(Cl)cn2)cc(Cl)ccc1Cl c1(-c2cn(CC(C)NC(c3ccc(O)nn3)=O)nn2)cccc2ncccc12 N1(C(c2cccnc2)=O)CC(F)(F)C1C1CCN(C(C2(F)CCOC2)=O)CC1 CN1CCN(C(=O)OC(C)(C)C)C(C(=O)Nc2ccccc2)C1=O.C1(=O)C(C)(C)N1 C12(CNC(CC(C)OC)=O)COC(CNC(=O)CCc3cc(C)[nH]n3)(C1)C2 C1(n2cc(CCCC(C)O)nn2)CC2CCC1(NC(C1CCC(C(N)=O)C1)=O)C2 C1(C(=O)NCC(N(C(=O)Cc2ccno2)C)C2CC2)CCCC(F)(F)CC1 Cn1cnnc1CCCC(=O)NC1COCC1NC(c1ccoc1C1CC1)=O C1(C(=O)NC2CCN(C(=O)CN3CCCC3CO)CC2)CCCC2(CC2)C1 CC(F)(F)C(C)(C)C(=O)NC1CS(=O)(=O)CC1NC(=O)C(O)(C1CC1)C1CC1 c1(COC)ccc(C(F)(F)F)c(C)c1.N12OCC(C1=O)NC2c1ccccc1 C(C)(C)(CC(=O)N(C)CCn1ccnc1C)NC(C1C(CC)CCO1)=O c1(C(N(C)CC2CCN(C(C(C)SC)=O)C2)=O)cc2ccccn2c1 Cn1cc2c(C(=O)NC3CN(C(C4CCCO4)=O)CC3F)cccc2n1 Cc1nc(O)nc(C)c1C(=O)N(C1CCCCC1)CCNC(C1CCC1(F)F)=O C(=O)(C(C)(C=C)CC)NCCCC(=O)N(CC(=C)CC)C.C1(=O)COCCN1 C1(C)(C(=O)NCC2N(C(CCSCCC)=O)CC2)CCN(C)C1=O C1(N(C)C(C2CSCN2C(=O)CCC2CCC2)=O)CCC(=O)NC1 c1(C(N2CCC(CCNC(C(C(C)(C)C)OC)=O)C2)=O)c(C)cc(O)cc1C C1(NC(C(C=CC)O)=O)CC2(CCN(C(c3cccc4nncn34)=O)C2)C1 c1(OC)ccc2nc(C)c(C(=O)NC(C)C(C)NC(c3ncoc3C)=O)cc2c1 C1(N(C(=O)CN2CCCC2)C)CCN(CC(=O)N2CCC2)CC1O C(CCC(=O)NC(c1n[nH]c(CO)n1)C)(C(C)C)NC(C(c1ccc(C)o1)C)=O C1(CC)(CCC=CCOC)CC1.C(C)(C)=CC(=O)NCCO.C1CO1.C(CO)O CC1CCCC(C)C1NC(c1cc(CNC(C2CCN2C)=O)ccn1)=O C1(C(N2CC3C(CNC(C4C(C)C4C)=O)(C3)C2)=O)CC2CCCC2C1 C1(C)(NC(C2C3N(C(c4c(C)nccn4)=O)C(CC3)C2)=O)CN2CCC1CC2 C1(C(C)NC(c2nc(C)oc2)=O)CCCCN1C(=O)Cn1cccn1 Cc1cnc2n1CCC(C(=O)NC1COCC1NC(c1cscc1Cl)=O)C2 N#Cc1ncc(Br)cc1NC(C1CN(C(c2ccc(F)c(I)c2)=O)CCC1O)=O CCCC(CNC(c1c(C)nsc1N)=O)C(=O)NC(c1nc[nH]n1)C1CC1 c1(Oc2cccc(CN(C)C(=O)Nc3ccc(Cl)nc3)n2)ccc(Br)cc1F CN1CC(C(=O)NCC2C(CNC(C3(C(c4ccccc4)=O)CC3)=O)C2)NC1=O C(CC(C(C)(C)C)NC(=O)Cc1ccsc1)N(C)C(C1CCCC1C1CC1)=O C1(CCCNC(COCC(C)(C)C2CC2)=O)CCCN1C(C1CC1(Cl)Cl)=O N1(C(CC2(C#N)CC2)=O)CC2CC1C2NC(c1sccc1F)=O CC1OC(C)CC1C(N1CCN(CCNC(C2COC(C)C2)=O)CC1)=O c1(NC2CC(NC(c3c(C)[nH]nc3Cl)=O)C2)ncnc2cccc(Br)c12 C1(C(=O)NCC=Cc2cc[nH]n2)CC12CCN(C(=O)CC1CC1)C2 c1(C(=O)NCCN2CCN(C(CCCC=C)=O)CC2)cnc2nc(Cl)ccc2c1 N1(C(c2cc(SC)c(F)cc2)=O)CCN(C(C2CC23CC(F)(F)C3)=O)CC(O)C1 N1(C(C)=O)CC2CCC(C1)N2C(c1cc2c(ccn2C)[nH]1)=O CP(C)(=O)c1cccc(=NCc2ccccc2N2CCCCC2)[nH]1 Cc1cc(C)nc(SCC(=O)NCC2CC2CNC(c2cc(Cl)c[nH]2)=O)n1 C1(C(N(C)CC2CCCN2C(C2(C)CCC(=O)N2)=O)=O)CSC(c2ccccc2)=N1 C1(NC(CCC)=O)CCCN(C(c2ccnn2C)C(=O)NCCC2CC2)C1 CCC(CC(=O)NC1CCOC1C(=O)NCCC(C)N1CCC1)OC c1(-c2cc(C(=O)NCC(CN(C(CC(C)N(C)C)=O)C)O)n[nH]2)cccc(Cl)c1 NS(=O)(=O)c1ccsc1C(=O)NCC1CCCC(NC(C2CC(F)(CO)C2)=O)C1 Cc1cccc2c1CC(C(=O)NCC1CN(C(C3(C)CCCCCC3)=O)C1)N2 C1(NCCNC(=O)NCC2(C(C)C)CC2)COC(C)C1 c1(N2CCCC(NC(C3(C)CC=C(C)CC3)=O)C2C)cc(C#N)ccc1[N+](=O)[O-] c1(C(N2CCCCC(NC(C3C(CCOC)C3)=O)C2)=O)ccc2nc(C)cn2c1 N1(C(c2c(CNC(C3CC(C)(C)C3)=O)ccs2)=O)CC2CC=CC1C2 C1(NC(Cc2ncc(CC)[nH]2)=O)CCCCN(C(c2c[nH]nc2F)=O)C1 N1(C(C2C(C)(C)CO2)=O)CC2CN(C(c3cccn4cnnc34)=O)CC2(C)C1 c1(C(=O)NCC2COCCN(C(C3(C)N(C)CCC3)=O)C2)coc(S(C)(=O)=O)c1 CCCCCCSCC(=O)NC1CC(C(=O)NC2CSC2)C1.n12cc(cn1)C2 C1(NC(C2C(C(=O)OC)C2)=O)CCN(C(=O)C(C)(C)NC(C)=O)C1 N1(CC)C(=O)NC(c2ccoc2C)C(C(=O)OC)=C1C1CCCCCCC1 COn1cnc(C)c1C(=O)NC(CNC(C1CC2(C1)CC(O)C2)=O)C(C)C C1(NC(c2cscn2)=O)(CF)CCN(c2ccnc(CO)n2)C1 C=CC(O)C(=O)NC(c1ccnn1C)C(=O)N(C)CCOC C1(CC(N2CC(CC(=O)OC)C2)=O)CC(NC(=O)CC2(C)CCOC2)C1(C)C N1(C(CCc2ccc(C)o2)=O)CCCC2(NC(c3cnn(C)c3F)=O)CC2C1 C1(NC(C(C)Sc2ccc(Cl)cc2)=O)CC2C1CCN2C(c1c[nH]nc1F)=O N1(C(CS(=O)(=O)NC)=O)CCC2CCCN(C(c3cc(Cl)c(N)cc3F)=O)C2C1 C1(CC(=O)Nc2cccc(C3CC3(F)F)c2)CCc2ccccc2C1 C12(C(N3CCC(CC)C3)=O)CC(CNC(=O)C(C)(C)F)(C1)OC2C Cc1cc(C(=O)N(C)CCNC(c2c[nH]nc2C2CCC2)=O)c(N)c(F)c1 CC(C)C(CN(C)C)N=c1[nH]c(=NCc2c(Cl)cnn2C)[nH]c2cccnc12 C1(C(N2CCC(NC(CCc3ccc(SC)cc3)=O)C2)=O)CN(S(N)(=O)=O)C1 c1(C(=O)NCC(C(C)C)(O)CNC(=O)C(F)(F)F)[nH]c2ccc(Br)cc2c1F C(=O)(N=c1ccn(CC2CC2)[nH]1)C1N(C(C)(C)C)CC(O)C1.N12CCC1C2=O C(=O)(C(C(C)C)NC(C)=O)N1CC(O)(CCNC(C(C)NC(COC)=O)=O)C1 C1(=CC(=O)NCCOCCCNC(C2C(C)OC(C)C2)=O)CCC(C)(C)CC1 N1(C(c2c(CC)non2)=O)CCN(C(=O)C2=CCC(C(F)(F)F)OC2)CC(O)C1 C12(C(N3CCCC3)=O)CCCN1C(=O)OC2.C(C)(C)(C)OCC N1(C(C(COC)OC)=O)CC(OC)CC1CCNC(=O)CCCn1ccnc1 CC1(C)CC(CC(=O)NCC2CCN(C(c3cnc(C(F)(F)F)s3)=O)C2)CCO1 O=C(C1=NOC2COCC12)NC1CN(C(=O)CCF)C2(CCC2)C1 C1(CCNC(C(C)OC)=O)CN(C(c2cc(-c3ccc(F)cc3)ns2)=O)CCO1 O(S(=O)(=O)c1ccccc1)c1ccc(N2C(=O)C(OC(F)F)CCC2)cc1 Nc1nc2c(cc1C(N1CC(CCO)C1)=O)CCC2.c12cn(nn1)CCCOC2 C1(CNC(CCCC(C)=O)=O)CN(C(c2cc(N)ccc2F)=O)C2CCCC2O1 c1(C(N2C(CNC(C(C)SCC)=O)C(CC)CC2)=O)nccc(N)c1Cl Cc1cc(C(=O)N(C)CC2COCCN2C(=O)CCCC2CC2)ccc1F C1(NC(C(C)=C2CCC2)=O)CCN(C(c2cccc(C3CC3)c2)=O)CC1C(C)C N1(CC(=O)N(C(CC)CF)C)CCCCC1c1nc(O)n[nH]1 C(=O)(C(C)(F)CCCC)N1CCC(CN(C(C(C=C)(C)C)=O)C)C1 c1(C(=O)NCC2CCC(NC(C3C(C)OC(=O)N3)=O)C2)ccc(C(N)=O)cc1F Cc1nccc(C(N2CCC(CN(C(=O)C(C)(C)c3ccns3)C)C2)=O)n1 C1(C(N(CCC(=O)NCC(c2nccs2)C)C)=O)CC1C1CCCC1 C1(N(C(=O)Nc2n(C)ncc2)CCOC(C)(C)C)CN(C(=O)CCCF)C2CC12 N1(CC(=O)NCCCCCNC(C2(Sc3ccccc3)CC2)=O)CCOCC1=O C1(C(N2CC(NC(c3coc4c3CS(=O)(=O)C4)=O)C2)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NCC(CN(C(c2cncc(OC)c2)=O)C)C)ccc2oc(C)nc2c1 N1(C(C(C)C#N)=O)CC(C(=O)Nc2cc(C#N)ccc2F)C2(CCC2)C1 c1(CNC2CC(NC(c3nn(C)c(Cl)c3)=O)C2)ncc(Br)cc1F CC(C(Cc1ccccc1)CO)NC(=O)CSCC(=O)OCC1CC1 CN1CCc2c(C(N3CCC4CN(S(=O)(=O)c5cnoc5)CC4C3)=O)cccc21 C1(OC)CC(F)CN(C(=O)CC2CCCN2C(=O)CC2(C)CC2)C1 N1(C(C(CC)OCC)=O)CCC(C(N2CC([N+](=O)[O-])C2)=O)(CC)C1 C1(=CCC(=O)NCCN(C(=O)C(C(C)C)C(C)(C)C)CCOC)CCC(C)CC1 c1(OC)ccc(NC(C2(NC(=O)CC3CCOC3)CCSC2)=O)cc1 N1(C(C(C)(C2CC2)OC)=O)CCC(CNC(c2c[nH]cc2C(C)(C)C)=O)C(C)C1 C1(C(N2CCOCC(F)(CNC(=O)CC3(CO)CC3)C2)=O)CCOCC12CCC2 C#CC1(C(=O)NC2CCCN(C)C2=O)CCN(C(c2c[nH]cc2C)=O)C1 c1(CN(C2CC(O)C2)C)ccc(O)c(-c2ccc(F)c(N)c2)c1 C(=O)(C(N=[N+]=[N-])C(C)C)N1C(C(N2CC(C(N(CC)CC)=O)C2)=O)CCC1 N(C1CC2(CN(C(c3c(C)cnn3C)=O)C2)n2ccnc21)C(C(C(=C)C)(C)C)=O Cc1cc(C(=O)NC2CC(CNC(=O)C(F)=C3CCC3)C2)c2[nH]cnc2c1 CC1(C)CN(C(c2cc(Cl)ns2)=O)CC(CNC(=O)Cn2cc(CO)nn2)O1 C1(C(=O)NCC(C)CNC(N)=O)CCCC(Nc2cc(C(F)(F)F)ncn2)C1 c1(C(=O)NCCCN(C(C2(C(C)C)CCCO2)=O)C2CC2)cnnc2ccccc12 C(=O)(C(=O)CC(C)CC)NC1CCCC(C(=O)NC(CC#C)CO)C1 c1(C(=O)NCC(CC)N(C(=O)C(O)CCC(C)C)C)c(C)cc(C)cc1C Cc1ccnn1C(C)C(N1CC=CC1C(=O)N(CC(O)CN(C)C)C)=O CC1CC(=O)NCCN1C(=O)COC1CC(NC(C2CNC(=O)O2)=O)C1 C=CCC(C)(C)CC(=O)NCC1CN(C(=O)COC2(C)CCCC2)CCCO1 C1(NC(=O)Cn2nccn2)C2CC3C(C2)C13C(N1CC(N(C)C)C(C(F)F)C1)=O c1(NC(C2CCCN(C(c3ncc(OC)nc3)=O)CC2)=O)nsc2ccccc12 Cc1nc2cc(C(=O)NCC(C)(CO)NC(=O)CC3CCC(=O)N3)cnc2[nH]1 Cc1cc(C(N2CCC(C(F)C(=O)Nc3cnc(CO)nc3C)C2)=O)ccc1O c1(N(C)C)ccc(CNC(=O)Cc2ccc(-n3cnnc3)cc2)cc1 C(=O)(C(O)CC[S+](C)C)NC1CC2C(NC(c3nccc(OC)c3N)=O)C2C1 C(N=c1nc(N2C3CCC2CC2(CC2)C3)c2c([nH]1)CCC2)c1ccn(C)n1 N1(C(C(c2ccc(CO)cc2)C)=O)CC2CN(C(c3cnn(C)c3)=O)CC2(C)C1 C#CC1(C(=O)NCCc2noc(=O)n2C)CCN(C(c2ncccc2F)=O)C1 c1(C(C)C)ncc(Cl)c(C(N2CCN(C(c3cc4ncsc4[nH]3)=O)CC2C)=O)n1 N1(C(=O)NC(C)C(c2ccc(Br)cc2)C)C2CCC1C(N)C2 c1(C(=O)NCC(N2CCC(Cn3cc(CCCC)nn3)C2)=O)ccc(C)cc1 CCC(C)C(O)C(C)C(=O)NC1(C(=O)NCCN(C)C)CCC(C)(C)C1 N1(C(c2c(CC)cccn2)C(=O)NC(C)CC)CC2CC(O)CC2C1 C1(NC(N(CCC)Cc2cccc(Br)c2)=O)CC2CC3C(C2)C13 N1(C(C2ON=C(CC)C2)=O)CCC(F)(CNC(C2(C)CC3CC3C2)=O)CC1 C1(C(=O)NCC(CC(=O)NCc2ncccc2Cl)C2CCC2)CC2(CCO1)CC2 c1(C(=O)NC23CC(NC(=O)COc4ccc(F)cc4)(C2)C3)ccc2nncn2c1 c1(N2CCC(NC(C)=O)C2)nc(N2CC3(C)COCC3(C)C2)nc2c1COCC2 C1(NC(CCC)=O)CN(C(c2ccccc2SCCO)=O)CC1OC N1(C(CN(CCCCCC)C)=O)CCC(CNC(=O)CC2OCCC2C)C(C)C1 N1(C(C(C)N(C)C)=O)CCN(C(c2ccn(CCO)c(=O)c2)=O)C(CO)C1 C1(CNc2c(C)c(Cl)nc(-c3ccccc3)n2)CC(=O)N2CCCCC12 C1(CCNC(CCN(CC)CC)=O)CN(C(=O)CC(O)CCSC)CCCO1 O=C(NNc1ncnc(Cl)c1Cc1ccccc1)C1CCCC(c2ccncc2)C1 Cc1nc(Cl)ccc1S(=O)(=O)NC(C1COCCN1Cc1cnc(N(C)C)nc1)=O S(=O)(=O)(c1ccc(N2CCCC(C(C)(C)C)C2)c(F)c1)NCCCOCC(C)C C(=O)(CCCC(CC)NC(=O)CC(C)OC(C)=O)N1CCC(OCC)C1 N1(C(C2N(C(c3ccc(C#N)[nH]3)=O)C(C3CC3)CC2)=O)CCC2C(C(N)=O)C2C1 Cc1nccc(C(=O)NCC2(C(=O)N(C)CC3CCCOC3)CCC2)c1N N1(C(C2ON=C(C)C2)=O)CCC(NC(c2cc(Br)no2)=O)C(C)(C)C1 CCCC1CCCNC(=O)COCC(=O)N1.C1(=O)CCCN1.C(C)(=O)OC(C)=O c1(C2(C(=O)NC3CC(CNC(CCCC=C)=O)C3)CC2)ccccc1C#N C(=O)(C(C)CC(C)C)NCCC1N(C(c2n(CC=C)ccc2)=O)CCSC1 C1(NC(c2c(CSC)cccn2)=O)CCCN(C(=O)CCC2CCN(C)C2)CC1 N1(C(c2n(CC)nnc2)=O)CC(C)(C)CC1CNC(=O)CC1CC(O)C1(C)C C(=O)(C(O)P(C)(C)=O)N(CCC)CCC.C(CC)NC(=O)COC(C)CC c1(N2CC(C)(CNC(c3c(OC)cc(Cl)nc3)=O)C2)ncc2cn[nH]c2n1 C1(NC(C(=O)NC(=O)C2CC2)CO)C2CC1N(C(=O)CCCc1cnn[nH]1)C2 Cn1cc(C(=O)NCCN(C(C2C3COCC23)=O)C2CC2)c(C(F)(F)Cl)n1 c1(C(=O)NC(CCCC)CNC(=O)CC2(C)CC(F)(F)C2)cc(O)nc(O)n1 Cc1nc2ccc(C(N3CC4CCCN(C(=O)CN(C)C)C4C3)=O)cc2o1.C(N)=O C1(CC(=O)NCC#CCNC(c2cnc(CCCC)s2)=O)CCCCC1F c1(-n2cc(COC3CCN(C(=O)C(F)CC4CC4)C3)nn2)ccc(F)c(Cl)c1 N1(CC(=O)NC2CN(C(CC3N(C(C)=O)CCC3)=O)C2)CCCC(O)C1 c1(CC)cc(-c2cc(C(=O)NCc3cc(C(F)(F)F)ccc3Cl)n[nH]2)ccc1C c1(C(N(C(C(=O)NCC(C#C)CC)C2CC2)C)=O)cccc(C)c1F N1(C(C2CN(C(c3c(CC)c[nH]n3)=O)C(C)CC2)=O)CC2CC(OC)C(C2)C1 C(COC)(C(=O)NCCCC1(NC(=O)Cc2c[nH]nc2C)CC1)OC.C(COC)O C1(C(=O)NC(C(CO)NC(Cc2c(C)cccn2)=O)C)COc2ccccc2O1 C1(N(C2(C(N)=S)CC2)C)CC2CC1CN2C(c1ccccc1)=O C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(c2ccc(CC)cc2F)=O)C=CC1 CC1c2ccccc2CC1C(=O)NC1(CO)CN(C(c2cc[nH]c2)=O)C1 C1(CC(N2C(CNC(CN(C)C3CC3)=O)CCC2)=O)Sc2ccccc2NC1=O N1(C(CC(=C)C)=O)CC(NC(=O)Cc2cncn2C2CC2)CC2(CC2)C1 c1(Nc2ccc(CN(CC)CC)cc2)nc2ccccc2n1C1CCN(C)CC1 CCC(CC)C(C(=O)N(C(C)C(N1CCC2CC1C(=O)O2)=O)CC)OC c1(OC)ccnc(C(=O)NCC(C)CC(=O)N2CCOC(CC(C)C)C2)c1 CC#CC1CCN(C(=O)C(C2CCCN(C(=O)CCCNC=O)C2)C)C1 N1(C(C=CC(C)C)=O)CCCC2C1CCCN2C(=O)C=CCN1CCC1 CC1=C(C(=O)N2CC(C(=O)NCC3(F)CCCCC3)CCC2C)CCC1 n1(CC(=O)NC(C2CN(C(C3CCC(F)(F)C3)=O)C2)C)ccc2ccc(F)cc12 c1(CNC(c2c(F)cc(F)cc2F)=O)nc(-c2ccccc2)n2ccncc12 C1(NC(C2CCCN(C)C2)=O)CN(C(=O)C(CO)NC(N)=O)CC12CCC2 C12(C(=O)NC3CCN(C(C(c4cc(C)oc4C)C)=O)C3C)CC1COC2(C)C CCCC(C(=O)NCc1nocc1C(N1CCOC(CC)C1)=O)NC(C)=O N1(C(CCC(C)=O)=O)CCC2(CC1)CC2C(=O)NC1COC(C(C)C)C1 CC(O)(CC(=O)N1CC2=C(C1)CN(C(=O)COCCCN=[N+]=[N-])C2)C(F)(F)F N1(C(C(C)S(C)(=O)=O)=O)C2CCC1CC(F)(CNC(=O)CCCNC(N)=O)C2 c1(C(=O)NC2C(CNC(C3(C)ON=C(C)C3)=O)C2)cc(O)nc2cnccc12 Cc1cc(N)ccc1C(N1CC(N(C)C(c2cnc(O)c(F)c2)=O)C2(CC2)C1)=O C1(CCC(=O)NCC(N2CCOCC2)CC)CCN(C(c2nocc2C)=O)CC1 C1(CNC(c2c(C)n(CC3CC3)cc2)=O)COCCN(C(=O)C2=CCCOC2)C1 Fc1ccc(-n2nc(CO)nc2-c2cnc[nH]2)cc1 c1(CNC(C2CCCN(C(c3ccn(CCOC)n3)=O)C2)=O)ccc(F)nc1C C1(NC(c2n(CC)nc(C(C)C)c2)=O)CN(C(=O)C(C)(C)OC(C)=O)CC(C)(C)C1 c1(C(N2C(C)CC(NC(=O)CC3CCCOC3)C2)=O)ccn2nncc2c1 N1(C(COCCC)=O)CC(F)(C(=O)NCC(C)OCCO)C1 c1(C(C2CC23CC3)NCC(C)CC2CC2)nnnn1C1CC1 C1(CNC(c2ccco2)=O)CCCN1C(=O)CNC(c1ccccn1)=O C(=O)(C1CCc2sc(NC(=O)N(C)CC3CCC(F)(F)C3OC)nc21)OCC CC(C)C(N=[N+]=[N-])C(=O)NCC1COC(CNC(=O)CCc2cncs2)C1 C1(NC(=O)Cc2cnns2)CCC12CN(C(c1cccn(C3CC3)c1=O)=O)C2 c1(OCC2NC(=O)CN(C(c3c(OC)cccc3)=O)C2)cc(C)c(F)cc1Cl c1(NC(C2C(C(=O)OCC)C2)=O)cc(Cl)c(C#N)cc1F N1(C(Cc2ncc(C)nc2)=O)CCC2CN(C(c3nccnc3Cl)=O)CC2C1 Cc1cc(CSc2nnc(-c3ccncc3)n2C)ccc1Cl N1(C(c2ccc(C)s2)=O)CCC2(CCOCC2)C(CNC(=O)C(C)CC(C)C)C1 C(=O)(CC(C(F)F)NC(=O)CCC(N)=O)N1CCC(NC(C)=O)CC1 c1(-c2ccc(C(=O)NC3CN(C(c4ccc(O)nn4)=O)C3)s2)ccc(F)c(F)c1 c1(CN(C2CCN(CC)C2)C(c2csc(C3CCCO3)n2)=O)ccc(F)nc1F c1(CCC)c(C(=O)NC(CNC(C2(C(=O)OC)CC2C)=O)CC(C)C)cnn1C C1(C(N(C2CC2)CC)=O)CC(=O)CC2CN(C(C3(O)CCC3)=O)CC12 c1(NC(C(C)(F)F)=O)ccc(C2=CCC(O)CC2)cc1F C(c1cccc(Cl)c1)=CC(=O)NC1(CO)CN(c2nc(C3CC3)ns2)C1 C1(NC(CCC2(NC(c3c(CC)nco3)=O)CCC2)=O)CCC(CC)CC1 c1(CNC23CC(NC(c4cc(Cl)nc(Cl)c4)=O)(C2)C3)ccc(C(F)(F)F)cc1Br C1(NC(c2ccccn2)=O)CN(CCCn2cncn2)CC1C1CCCC1 Cc1nn2c(C(N3CCC(CNC(c4ncccc4Cl)=O)C3)=O)c(Cl)nc2s1 c1(CNC(c2scc(-c3ccc(OC)cc3)c2)=O)cc(C)nc(Cl)c1 C(=O)(C(C)C(=O)N1CCOCC1CC(=O)NCC1(c2ccccc2)CC1)OC C(=O)(CC(C)CC(=O)NC(CC1CC1)C(=O)Nc1cccc(F)c1)OC C1(CC(=O)N(C2CCN(C(C=CC=CC)=O)C2)CCC)SC2=NCCN2C1=O C(=O)(CCCn1cc(CCC#N)nn1)N(C(C)(C)C)CC(=O)O c1(CNC(C2(C)CC=C(C)CC2)=O)nc2c(s1)CN(C(c1ccoc1)=O)CC2 N1(C(CC=C(C)C)=O)CC2C(NC(C3(C4CCCO4)CC3)=O)C2C1 C1(NC(CCc2cccc(C)c2)=O)CCC(C)N(C(=O)C(F)=CC2CC2)C1 C(=O)(C1CCCn2c(CC)nnc21)NC1CC(CNC(COCCC)=O)C1(C)C c1(C(=O)NC2(C)CCN(C(C34CCC(CC3)CO4)=O)C2)cc2ccc(Cl)cc2o1 N1(C(CCCN(CC)CC)=O)CC2(CC(NC(C3CCN(C)C3C)=O)C2)C1 C1(C(=O)NC(CNC(C2(C(C)C)CCC2)=O)(C)CO)CS(=O)(=O)CC(=O)N1 CC(C)(C)C(=O)C(=O)NCCOC1CCN(C(=O)C(O)CN2CCOCC2)CC1 C1(CCOC)(C(N2CCC(O)(CCNC(=O)C(C)(C)CF)C2)=O)CCN(C)CC1 S(=O)(=O)(c1cc(C(C)C)ccc1NC1CSCC1C)N1CC2(CC(OCC)C2)C1 C(=O)(C(CC)C(=O)N(C1CCCCC1NC(=O)C(F)=C1CCC1)C)OCC N1(C(c2cn(CCOC)nc2)=O)CC2C3CCC(C2C1)N(C(C1(CO)CC1)=O)C3 CCC(C)(C)CC(C(=O)NCCCF)N1CCOC(C(N)=O)C1 C=CC1(C(=O)NC2(C(=O)O)CCC2)CCC1 C1(C(N2CC(NC(C(C)(C)N(C)C)=O)C(F)CC2)=O)Cc2ccccc2C1 C=CCC(C)(O)C(=O)NOCC(=O)NCCC1COC(C)(C)C1 C(=O)(C(C)N(OC)C(=O)C1COCCC1NC(=O)CC12CCCC1C2)OC C=CCC1C(=O)NCCCC(=O)N1.c1(CNC(C)=O)nnc(C)n1CC c1(C(N2CCN(Cc3ccc(C)cc3)CC2CC#N)=O)cccc2ccnn12 C(CNC(=O)C(Cc1ccccc1)N(C(=O)CCOC)C)(CC(C)C)OC c1(C(N2CCC(NC(COC(C)=O)=O)C(C(C)C)C2)=O)cc2cccn2c(O)n1 CC(C)C(CCc1ccccc1)(c1nnnn1C)NCC1C=CCCCC1 N1(C(c2cc(C)cc(Br)c2F)C(=O)NC(C(=O)OC)C)CCc2ccc(F)cc21 N1(C(C(C)Cn2ncc3ccccc23)=O)CCC(F)(F)CC12CCC2 N1(C(COCC)=O)CCC(C)(C)CC1C(=O)Nc1cnc(CC)nc1C C(CN=c1[nH]c(=NCC2CC23CC3)[nH]c2c1CSC2)c1n(C)c2c(c1)cccc2 CC(C)(O)C(O)CNC(=O)CCC1CC(NC(C2C3CC(CC3)C2)=O)C1 c1(C(C)=O)ccc(CC(=O)NCCC(C)(C)NC(=O)C(=Cc2cccs2)C)cn1 CCCCCCC(C)C(=O)N(C1CCN(C(c2cnc(C3CC3)s2)=O)CC1)CC C12(NC(C(CCCC)F)=O)CCCC1N(C(c1nc(C3CC3)cs1)=O)CC2 C=Cc1cc(C(=O)NCC2(NC(=O)C(CN(C)C)CC)CC2)cc(F)c1 N1(C(CS(=O)(=O)NC)=O)C2CCC1CC(CN=c1ccnc(C3CCC3)[nH]1)C2 Cc1ccc(OC(c2ccc(C3CCOC3)cc2)=O)c(C(C)C)c1 CC1CCCC(CC(N2CCC(CC(=O)NC34CCN(CC3)C4)C2)=O)O1 C1(C(N2CC3C(CNC(c4nccc(C)n4)=O)(C3)C2)=O)CC(C2CCC2)C1 C1(NC(CCCOCCC)=O)C2CCC1N(C(=O)CC1CCCCN1C)C2 c1(CNC(=O)C(O)CC2CCCCC2)cccc(NC(C2CCC3(CC3)C2)=O)c1 C(CCNC(C1COCC1C(N)=O)=O)(CNC(=O)C(C)c1ccco1)OCC CCC1=NOC(C(=O)NC2(CNC(c3cc(C)c(C)[nH]3)=O)CCC2)C1 c1(OC)ccc(C(C)=CC(=O)NCCN(C(=O)CSCC(C)C)C(C)C)cc1 C1(OC)(CNC(c2csc(-c3cnn(C)c3)n2)=O)CCN(C(=O)CNC(N)=O)C1 C1(n2cc(CNCc3cc(COCC)no3)nn2)CCCC(C(=O)O)C1 c1(N(C2CCC2)CCNC(c2nc[nH]n2)=O)nnnn1CC1CC1 Cc1cnccc1N1CCN(C(=O)NC(c2ccc(Br)cn2)C(F)(F)F)CC1 CC(CC(=O)N1CC(S(C)(=N)=O)C1)CC(C)(C)C.C1(CCOCCO)C(=O)N1 c1(C(N2C(CNC(C(C)S(N)(=O)=O)=O)CC3CC32)=O)ccc(F)c(O)c1F C(=O)(C(C)(O)CC(C)C)NC1C(NC(C2CCN(CC(C)C)CC2)=O)CC1 c1(CN2C(C(=O)NC3CC3c3ccc(F)cc3)CC(O)C2)cc(I)ccc1O Cn1nnc2c1CC(C(=O)NCC1(O)CCCN(C(C34CC(C3)C4)=O)CC1)CC2 CC1CC(CN)C(C)CN1C(=O)COCc1cccc(N(C)C)c1 C(N=c1[nH]c(=NCCNS(=O)(=O)N(C)C)[nH]c2c1COCC2)C1C(SCC)C1 C1(F)(C(=O)NC2CC(NC(C3CCC(C)CC3)=O)C2)CCCN(C)C1 CCS(=O)(=O)N1CC(C(=O)NC(C)C(c2cccs2)NC(=O)CCOC2CC2)C1 C(=O)(CCCS(C)(=O)=O)N1CC(NC(c2ccn(C(C)(C)C)n2)=O)C2C1C2 C1(C(N2C(CNC(C=Cc3nc(C)c(C)[nH]3)=O)CC2)=O)CC2OC(=O)OC2C1 c1(C(=O)NCC2(NC(C3C4CC(F)(F)CC34)=O)CCOC2)cc2ccncc2[nH]1 C(=O)(C(CC(F)F)NC(C1CS(=O)C1)=O)NCC(C)(O)CO C1(=O)CC(C)NC(=O)COC(C)(C)CN1CC.C(=O)(CCC1CCCO1)OCC C1(C(N2CC(OC)C2)=O)C(C)CCN1C(c1cnccc1C)=O c1(C(N2CCN(C(=O)Cn3ccnn3)C(C(F)F)C2)=O)cnc2ncccc2c1 c1(OC(C)C(=O)NC(C)(C)Cc2ccc(I)cc2)ccc(Cl)c(F)c1 C#Cc1ccnc(C(N2CCCC2CN(C)C(C2C3C4CCC(C4)C23)=O)=O)c1 n1(CC(=O)NCCN(CC(C)O)C(C2CCCSC2)=O)cc(C#N)c(O)nc1=O Cc1cc(=NCC2(S(N)(=O)=O)CC2)[nH]c(=NCC2CCCCN2CCN(C)C)[nH]1 N1(C(CC(C(F)F)NC(COCCOCC)=O)=O)CCC12CCOCC2 C1(C(=O)NCC(CNC(c2ccc(C(F)F)nc2)=O)F)CCc2nc(O)[nH]c2C1 c1(C(=O)NCC(C(C)C)NC(C2CCOC2C)=O)cc(F)c2[nH]nnc2c1 C1(CNC(c2ccc(O)cc2)=O)COCCN(C(=O)CC2CCCC2)C1 C1(NC(c2ccn(C(F)F)n2)=O)CCOCC1NC(C1CC(CF)C1)=O CC(C)C(=O)C(=O)N1CC2C(CNC(c3cccnc3)=O)C2C1 C=C1CCN(C(c2ccsc2)=O)C(C(=O)NC2CC2C2CC2C)C1 c1(C(=O)NC2CCN(C(C3(CN(C)C)CC3)=O)CC2)ccc(S(C)=O)cc1 c1(C(=O)NCCC2CCC(NC(C34CCC3CC4)=O)C2)ccc(F)c(F)c1 c1(C(=O)NC2CN(C(c3ccc(C(OC)OC)o3)=O)C2)nccc2n[nH]cc12 C1(CN(C(CC2CC(C)C2)=O)C)CN(C(=O)C(F)(F)c2ccnn2C)CC12CC2 C(CN=c1[nH]c(=NCC2CC3CCC(C2)S3)c2cc(Cl)ccc2[nH]1)CCN(C)C CC1CN(C)CCCN1C(C1(CO)CCN(C(c2cc(Cl)co2)=O)C1)=O C12CCC(CC1)CNC(=NC)N2.N1(C2CC(OCCOC)C2)CCCC1CO C1(NC(CC2(CC)CCC2)=O)CC(C(=O)NC2CC2CCOC)CC1O CN1CCCCC1C(=O)NOCc1ccc(Oc2cccnc2)cn1 C1(C(=O)NC(c2c(C)ncs2)C)(NC(=O)CC2CCCC3CC23)CCN(C)C1 N1(C(=O)CCCOC2CC=CC2)CCN(C(C2CC(O)C2)=O)C2CCCCC2C1 C(=O)(C1CCCc2ncnn21)N(C(CC)CNC(=O)Cn1ccc(C)c1)C N1(C(c2cc(OC)no2)=O)CC(C)C(C)(CNC(c2[nH]cc(C)c2C)=O)C1 C1(NC(Cc2c(CC)n[nH]c2CC)=O)CCN(C(c2cnoc2)=O)CC(C)(C)C1 C1(CNC2C(C)CC2)C=CC2(CCCCCC2)CC1 Cc1ccccc1-c1csc(CNC(=O)NCC2CCC(C(F)(F)F)O2)n1 C1(C(=O)NC2C(NC(c3cn(C4CC4)nn3)=O)COCC2)COCC2(CCC2)O1 C1(C(N2CC(=C)C2)=O)CCC(SC2CC2)N1C(=O)Cc1cnns1 C1(C(N2CCC(N(C(CCCN=[N+]=[N-])=O)CCO)C2)=O)CCn2cncc2C1 c1(C(=O)NCC(CN(C(=O)CC2CCCN(C)C2)C)O)cccc(CF)c1 Cc1c(Cl)c(C(=O)NC2(CNC(C34COC(CF)(C3)C4)=O)CCOC2)nn1C Cc1cc(Cl)c(C(N2C3CCC2CC(NC(C2(C(C)C)COC2)=O)C3)=O)cc1C N1(C(c2cc(CCC)nn2C)=O)CCN(C(C2(CC)CCCC2)=O)CCC1C CC(=O)CCCC(=O)N1CCC(C)CC1CNC(c1cc(F)n[nH]1)=O Cc1cccc2c1C(C)CC2CC(=O)NCC1(CNC(c2cc[nH]n2)=O)CC1 N1(C(CSCCOC)=O)CC(NC(c2c[nH]c(Br)c2)=O)C2CC12 c1(C(=O)NC(CC)CNC(=O)C(O)C2CCCC2)cccc(C(OC)OC)c1 n1(C(C2CCCCC2)C)nc(-c2cccs2)nc1-c1ccon1 CC1CN(C(C2(C)CC3CCC2C3)=O)CCC1NC(C1CC2CCC1C2)=O c1(C(N2CCCN(C(c3cnc(C)n3C)=O)CC2C)=O)cnn2c1C(=O)CCC2 N1(C=O)CC2CC(CO)CC2C1.C1(C2C(COC)(CN)C2)C(C(=O)C(=O)OC)C1(C)C Cc1cc(F)c(CN2C(C(=O)Nc3cnn4cccnc34)CCC2C)c(F)c1 n1(CC(C)C)ncc(C(=O)NC(C)C(C)NC(C2(c3cccnc3)CC2)=O)c1N C1(NC(C(CCC)F)=O)CCCN(C(c2cccc(F)c2N)=O)C1C c1(C(N(C2CCN(C(=O)Cc3nnc(C)o3)C2)CC)=O)ccnc2ccsc12 c1(C(N2CC(O)(c3nccs3)C2)c2ccsc2)cccc(Cl)c1 c1(CSCC(=O)NCC2CC(NC(=O)CCc3cc(Cl)cs3)C2)ccc(F)cc1 N1(C(C(N)Cc2csc3ccccc23)=O)CC2(CCC2)CCC1CO C(=O)(C(C)(C)CNC(C1CC2(CC2)C1)=O)N(C)Cc1c(C)ncs1 C(=O)(C(C)=Cn1ccnn1)NCC1CC(F)(CNC(C=C(CCC)C)=O)C1 N#Cc1ccc(C2(O)CN(CC(=O)Nc3nc(-c4ccc(OCF)cc4)cs3)C2)s1 c1(C(=O)NC2CCC(NC(=O)C(O)C3CCC3)CC2)c[nH]c2ncnc(O)c12 C1(CN(C(CCN(CC#C)C(C2(C)CCC(=O)N2)=O)=O)C)C(C)(C)C1(C)C c1(C(=O)NC2C(NC(C3(CC)CC3)=O)CS(=O)(=O)C2)cccc2c1oc(=O)n2C C1(NC(c2c(C)noc2)=O)CCCCN(C(C2CCC2)=O)C1 N1(C(c2nnc(C)s2)=O)CCOC(CNC(c2c(C)nsc2Br)=O)C1 Cc1sc(C(=O)NC2CC(NC(c3cc(C(F)(F)F)nc(C)n3)=O)C2)c(C)c1C c1(CNC(C(CNC(C2C(CC)CC2)=O)O)=O)ccc(C)c(O)c1 n1(CC)cccc1C(N1CC(C(=O)NCCNC(=O)C(N2CCNC2=O)C)C1)=O CC(C)CC(O)C(C)C(=O)NCc1cccnc1C(N1CC(O)CC1(C)CO)=O N1(C(c2nc(OCC)oc2)=O)CCC2CCN(C(=O)CC3CSC3)CC12 c1(C(N(CC(F)(F)F)CC2(NC(C(=O)OC)=O)CCCSC2)=O)cc(Cl)c(C)cn1 CC1OC2(C)CC1(C(=O)NC13CCC1CN(C(c1ccc(N)c(Cl)c1)=O)C3)C2 c1(C2(NCC3N(C(=O)OC(C)(C)C)CCCC3)CCC2)cccc(C(F)(F)F)c1 N1(c2nnc(C(C)SCC(F)(F)F)n2CCCN(C)C)CCC2C(C1)C2(F)F C(=O)(C1=NN(CCO)C(=O)CC1)NCC1N(C(C2(C)CCCS2)=O)CC2(CC2)C1 C1(NC(c2cnc(CC)o2)=O)CC(NC(C23CCC(CC2)C3)=O)C(O)C1 C1(C(=O)NCC2CC(NC(CC(C)CN(C)C)=O)C2)CCC2(CCCC2)C1 C1(C(=O)NC(C#N)C(N)=O)CC2(CC2)CN1Cc1ccc(O)cc1Cl N1(C(C(C2CCC2)OCC)=O)CCCN(C(c2cnc3nccn3c2)=O)C(C)C1 c1(OCC(=O)NCc2cn(C(CCCC)CC)nn2)ccc(F)cc1N c1(C(=O)NCCOC2CCN(C(c3c(CC)nc[nH]3)=O)C2)ccc(C)nc1O C1(CC)C(NC(=O)COc2cccc(O)c2)CCCN1C(=O)CC1CC1CC CC1=C(C(=O)N2CC3CN(C(=O)CC(C)C(C)C)CC3C2)COCC1 N1(C(=O)Nc2n(CC)nc(C(F)(F)F)c2)CCc2cccc(O)c21 O=S(=O)(c1cccc(NCCS(=O)C(F)(F)F)n1)NCc1ccc(Cl)c(F)c1 C1(O)(C(C)NC(C=CCCC)=O)CCN(C(=O)CC2CCC(C)CO2)CC1 Cc1cc(C(=O)NC(C(N2CC3(CCCO3)C2)=O)c2ccco2)ncc1N C1(C(C)(C)C)(CO)CCCN(N2CC3ON=C(CC(F)F)C3C2)C1 c1(C(=O)NCCC2(O)CN(C(C3N(C)CC(O)CC3)=O)C2)ccnc2c1CCO2 C(=O)(C(C)CC(C)C)N1C(CNC(c2n(CC)cnn2)=O)CC(OC)C1 C(C)(C)(C(C)N(C(=O)CCc1nc(C2CC2)no1)CC)NC(C(=O)NCCOC)=O C(=O)(C1CC(C)(C)Oc2ccccc21)N1CC(CCNC(C(COC)OC)=O)C1 c1(C(=O)NC23CCN(C(c4c(C)nc[nH]4)=O)CC2C3)cc2c(o1)CCCNC2=O c1(C(=O)O)ccc(CNC2CCC(N3CCOCC3)C2)cc1 C1(C(=O)NC(C)CSC(F)F)CCCCCC1NC(c1cc(O)nc(O)n1)=O C(=O)(CCCC(F)(F)CO)N(C1CCCN(C(=O)CC2CCC(C)C2)C1)CC c1(C(C)OC)nc(C)c(C(=O)NCC(C)N(C)C(c2cnc(C3CCC3)s2)=O)s1 c1(NC(C2CCCN(Cc3ccc(Br)cc3)CC2)=O)cc(F)c([N+](=O)[O-])cc1F c1(C(=O)OC)ccccc1N(C(=O)CSC)CCOCCO.C(CN(C)C)O c1(C(N2CCC(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)c(Cl)nn(C)c1Cl C1(NC(C2N(CCOC)CCC2)=O)CC2CC(C1)N(Cc1csc(C(C)C)n1)C2 c1(C(N2C(CN(C(C=COCC)=O)C)CCCC2)=O)c(F)ccc2n[nH]cc12 N1(C(C2CC(C#N)C2)=O)CC(F)(F)CC1CCNC(=O)CC1C=CCC1 c1(CC(=O)OC)c[nH]c(C(=O)N(CCCCN(C)C(C2CC=CCC2)=O)C)c1 N1(C(CC(C=C)C)=O)CCC2(CC2NC(c2cc(C3CC3)no2)=O)C1 c1(OC)ccccc1C(CNC(C1CC1CF)=O)NC(=O)Cc1nc(C)sc1C c1(OC)cc(CNc2ccc(C(=O)Nc3nc(C)cs3)nc2)ccc1C c1(CCNC(C(c2cc(C)n(C)n2)N)=O)ccc(Cl)c(C(=O)O)c1 C(CC(C)(C)CNC(C1C=CCN1C(=O)C(C)NC=O)=O)OC N1(C(=O)OC)CCCC(CC(N2CC3CC3(NC(C3CC3C(C)(C)C)=O)C2)=O)C1 Cc1cc(S(=O)(=O)NC(N)=O)ccc1C(F)(F)C(F)(F)F C#Cc1ccc(C(=O)NCC2CCN2C(=O)C(C)N(C)C(C)=O)cc1 N1(C(CC2(C)CCCO2)=O)CCC2(CCN(C(c3cnc(N)c(Cl)c3)=O)CC2)C1 c1(CCC(=O)N(C(CNC(CC2C(=C)CC2)=O)C)CC)cc(Cl)cs1 CS(C)(=O)=NC(=O)CNC(=O)NCc1ccc(F)c(F)c1Br N1(CCCC2CC(C(=O)NC(C3(C=C)CC3)=O)CO2)CCCC(O)C1 c1(SCCNC(C2C(CNC(C(C3CCCO3)OC)=O)C2)=O)n[nH]c(C)n1 c1(NC(=O)Nc2cnc(-c3cccc4c3CNC4=O)[nH]2)ccc2c(c1)C(=O)NCC2 C1(C2CN(C(C3CC3Cl)=O)C2)(NC(C2CCCCC2)=O)CC1 C1(CNC(c2cnc(COC)s2)=O)CCN(C(=O)C(c2cccnc2)OC)CC1 CCCC(C(=O)NCC1C2CN(CC(C)O)CC12)S(N)(=O)=O CC1C(NC(=O)C=CC2CCCO2)CCN1C(=O)COc1ccc(Cl)cc1 c1(N(C(=O)CN2CCCC2)C(=O)NCC)cccc(F)c1N c1(CCC(=O)NCCCN(C(C2C(SCC)C2)=O)C(C)C)cc(C(C)=O)c(C)o1 c1(C(N2C(CNC(C(CCCOC)C)=O)CC(F)C2)=O)cc(C)c(O)c(C)c1 C(CCC)(CCCNC(=O)C(F)=CCCF)NC(C(C)SCC)=O N1(C(CCSCCCC)=O)CCN(C)CC1CNC(C1CC1(Cl)Cl)=O N1(C(CC(CCSC)O)=O)CC(CNC(=O)CN2C(=O)CCC2=O)CC12CCC2 c1(C(=O)NCCC(=O)NCc2c(C(C)C)ocn2)cnn(C)c1N c1(C(N2CC(O)CC(NC(C3CC4(CSC4)C3)=O)C2)=O)c(Cl)ccc2ccoc12 C=CCCC(C)(C)C(=O)NC(C)CC(C)NC(C1(c2cc[nH]n2)CC1)=O N1(C(C2(OC)CCCOC2)=O)Cc2[nH]nc(C(N3CC=CC3CN(C)C)=O)c2C1 c12cccc(c1)NC1(CC1)CNC2=O.C(C(=O)N(C)C(C)C)OCCOC N1(C(=O)CCNc2ccccn2)CC2CCCN(C(c3cnc(CO)s3)=O)C2C1 Cc1cc(Cl)c(C(=O)NC2CN(C(=O)C(C)n3ccnn3)CC2O)cc1C C1(C(=O)N(C2CCCC2)CCO)CCCN(CC(=O)NCCCOCC(F)(F)F)C1 Cc1cc(CN(C)CC2CCN2C(=O)CC2(C)CCC2)n(C)n1 CC1NC(=O)CCC1CNC(C1CCN(C(C2CCCCC2)=O)CC1)=O CC1OCCC1C(N1CCC(CC(=O)NCC2CC(F)(F)C2)C1)=O C(C(C)(CC(=O)O)NC(=O)COc1ccc(C(=O)O)cc1O)OC c1(C(=O)NCCC2CC(C(=O)NC(CSC)(C)CO)C2)nc(C)ccc1C C#CCCCC(C)C(=O)N1CC2CCC(CNC(=O)COCC3CCOC3)C2C1 CC1CC(NC(=O)C=CC2CCCN2C(=O)CCN2CCCCC2)CCC1(C)C C1(C(=O)NCC2N(CC)CC2)CN(C(c2ccoc2)=O)CCC1(C)C C1(C(=O)NC(C2CCN(C(Cc3cc(CC)no3)=O)C2)C)CCC(N=[N+]=[N-])CC1 c1(-c2cccc(C(=O)NC3(CCCC)CCC3)c2)ccccc1S(=O)(=O)N(C)C Cc1ccc(-c2cc(C)on2)cc1.C(=O)CCN(C)C(C)=O.C12CC1COC2=O c1(-c2cc(C(=O)NC3C(NC(C(CSC)O)=O)C3)on2)ccc(Cl)cc1 N1(C(C(N2CCN(C)CC2)C)=O)CCC2(NC(c3ccccc3Cl)=O)CCCC12 S(=O)(=O)(c1c(F)cccc1F)N1C(C(N2CC(O)C2)=O)CC(F)C1 CC(CCCN=c1nn[nH]n1Cc1ccccc1)NC(C1(C)CC(=O)C1)=O C1(CN(C=O)Cc2cccc(OC(F)(F)F)c2)CC2OCCC2O1 c1(NC(=O)C(=O)NC2CCOC2)cc(NC2CC3CCC2C3)c(Br)cn1 c1(C(N(C2CCN(C(c3nc(CCC)oc3)=O)C2)CC)=O)nnn2c1CCC2.OCC N1(C(c2c(F)ccc(OC)c2)=O)CCCCC(NC(=O)CC(C)SC)CC1 c1(C(=O)NC2CCCN(CCNC(N3CCCCC3)=O)C2)nnn2c1CCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CC23CCCC2(C1)CN(C(=O)CSC(F)(F)F)C3 C(=O)(CC(C)(C)C(F)F)NCC1CC(C)N(C(=O)Cc2ncsc2Cl)C1 C1(SCC)CCC(C(N2CCC(NC(C3CC3)CC3(C)CCC(C)C3)C2)=O)CC1 Cc1cccc2c1CCOC2C(=O)NC(C)C(CO)NC(c1ccc(N)cn1)=O Cc1c(C)n(C)c2ccc(C(=O)NCC3(O)CN(C(C4(F)CC4(F)F)=O)C3)cc12 C1(COC)(CNC(c2n[nH]c(C)c2C)=O)CCCN1C(c1[nH]cnc1C)=O Cc1cc2[nH]c(C(=O)NC3C4CC3CN(C(c3ccc(F)cc3Cl)=O)C4)cc2o1 C=CC1OCCCC1C(=O)NCCC1CCN(C(=O)C=CCO)C(C)C1 CCC(CCC(=O)NC(C(=O)Nc1cccc(OCF)c1)C1CCC1)OC c1(SC)nc(N2CCC(NC(C3(C)CCC3)=O)C(C)C2)cc(Cl)n1 C(CC(=O)NC(c1cncs1)C)(CC(C)C)NC(c1c(C)nncc1)=O C(c1ccc(C(=O)NC2CCC2NC(C2CCC(=O)NC2)=O)o1)=CC(=O)OC c1(OC)ccc(CCNC(Cc2ccccc2)C(C)C)c(F)c1 C=CCC(C)C(=O)NCc1ncoc1C1CN(C(c2ccc(OC)o2)=O)C1 c1(NC(C(N2CCN(C(C3CNC(=O)N3)=O)CC2)C)=O)cncc(N)n1 CC(C)(C(=O)N1CC2(CCC(CNC(C3(C)CCOC3)=O)O2)C1)S(C)(=O)=O c1(C(=O)NC(CNC(C(C)NS(C)(=O)=O)=O)(C)C)ncc(F)cc1N c1(CC(=O)N(C2C(N(C(=O)C(O)C(F)F)C)CCCC2)C)ccn2cncc2c1 C1(CNC(c2cnc(CC)s2)=O)CCN(C(C2CC2c2cccnc2)=O)CC1C C=C1CC2(C1)C(=O)NC2.C(=O)(C(C)CN(C)C(C)=O)NC1CC(n2cncn2)C1 Cc1csc(N2CCCC2C(=O)NCC(C)NC(=O)C(F)(F)C2CCCCC2)n1 c1(C(C(=O)NC2C(NC(C(CSC)(C)C)=O)C2)C)ccc(F)c(Cl)c1 Cc1nc(C)n(CCCC(=O)NCCC(C)NC(=O)CN(C)C(C)C)n1 c1(C(N(C2(C(=O)NC(C(=O)OC)CCF)CC2)C)=O)cc(C)nc(C)c1 BrC1=CC=CCC2C3(CCOC1CNCCC2)CC3 C1(CNC(CCC#C)=O)COCC2(CCN(C(C3(C)CCN(C)CC3)=O)CC2)O1 c1(OC)cc(C(=O)NCCC2CN(C(=O)CNS(C)(=O)=O)CC2C)c(Cl)cn1 CC(C)(O)C(C)(O)CNCC1CC(C(F)(F)F)CO1 CC(F)(F)C(C)(C)CC(=O)N1CCCOC(CNC(C2CCCN2C=O)=O)C1 N1(C(c2cnc(C)nc2C)=O)CCOC2(CCN(C(=O)C(C)(C)Br)C2)C1 Cc1c(C(N2CCC(CCCNC(=O)C(CO)NC(N)=O)CC2)=O)ncn1C C1(CC)CN(C(c2ccc(OC)nc2Cl)=O)CCN1c1ncccn1 CC1CCCCC1C(=O)NC1(C)CCN(C(C(=O)Nc2cn(C3CC3)cn2)=O)C1 c1(C(=O)NCC23C(CN(C(C(C)=O)=O)C2)C3)cc(SC)ccc1[N+](=O)[O-] c1(C(C(=O)NCC(=C)C)N(C(C)C)C2CC2)cncn1C N1(C(c2cccc(C)c2)=O)CCC(C)C(NC(=O)CC2SC3C=CC2CC3)C1 CC(C)(CNC(C1CCCO1)=O)CCNC(c1ncoc1C1CC1)=O C#CCC(C(=O)NC(CCF)C(=O)NC(c1ncc(C)cn1)C)C1CC1 c1(C(=O)NC(CC)(C)CNC(C2CC2C(C)(F)F)=O)cncc(C#N)c1 C12(NC(c3c(C)cccc3Cl)=O)CCCN(C(C3CCCC(=O)N3C)=O)CC1C2 C(=O)(C#CC(C)(C)O)N(C)CC1CCCCN1C(c1cn(C(C)(C)C)nn1)=O c1(C(N2C(CNC(C3(COC(C)C)CC3)=O)CCC2)=O)ccc2nnc(O)n2c1 C(N=c1[nH]cnc(Cl)c1OC)C1CCCC(NC(CC(C)SC)=O)C1 c1(C(=O)NCC2(C)CCN(C(C3CC3(C)C(F)(F)F)=O)C2)ccc([N+](=O)[O-])o1 C1(C)(C2C(=C)C2C(=O)NC2CCCC(NC(=O)NCC)C2)CC2(C1)CC2(F)F c1(C(N2CC(C(C)NC(C(C)OCC)=O)C2)=O)cc(C#N)c(F)cc1F C1(NC(C=CSC)=O)(CNC(=O)CCC2CCCC(O)C2)CCCCC1 C1(C(=O)OC)COCC1Cn1cc(CCS(N)(=O)=O)nn1 c1(C(N2C(C(=O)NC(c3nccs3)C)CC(O)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] N(C(=NCCc1ccsc1)NCC(F)F)Cc1n(C)nc(CO)n1 C(=O)(CC(C)C(F)(F)F)N1CCC(OCCNC(C2(COC)C=CCC2)=O)C1 CCCC(O)C(CO)NC(=O)C1=CCN(C(c2n[nH]c(C)c2C)=O)C1 N1(C(c2nn(C)c(C3CC3)c2)=O)CC(NC(=O)Cn2cnnc2)C2CCCCC12 N1(C(c2c(CC)n(C)cc2)=O)CC2CCCC1CN(C(c1cc(C)oc1C)=O)C2 C1(NC(C2C(C)C2C)=O)CC2(CCN(C(C3C4CCCCCCC34)=O)C2)C1 N1(C(Cc2ccn(C)n2)=O)CCn2cc(C(=O)Nc3ncc(CCO)s3)nc2C1 N1(C(CC2(OCC)CC2)=O)CC2(C)CN(C(C3(C(F)F)CCCC3)=O)CC2(C)C1 N1(C(CCC=C(C)C)=O)CCC2(C1)CN(C(c1cn3c(n1)CCC3)=O)CC(C)O2 N1(C(C(C)C2CC2)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C12CCC2 N1(C(c2cc(Cl)ns2)=O)CCC2(C1)CN(C(=O)CCc1ccc[nH]1)C2 C1(NC(=O)Cc2cc(Cl)cs2)CC2CCC1(NC(=O)CC1(O)CCCC1)C2 N1(C(C(=O)NCC#C)C)CCC(NC(=O)OC(C)(C)C)CC1.n12cc(cn1)CC2 C1(CC(=O)OC(C(=O)OCCOCP(C)(C)=O)=O)COCCN(C(C)(C)C)CO1 c1(C(=O)NC2CCN(C(c3cnc(S)nc3)=O)CC2)ccc(Br)cc1F Cc1ccc(CC(=O)NCC2C3CN(C(=O)C(C)(C)CO)CC23)cc1Br CCC(CCC(=O)N1CC(Cn2cc(-c3cncs3)nn2)C1)OC c1(CNCc2cc(Br)sc2)cc(N2CCCC2)ccn1 C(CCN=C(NCCCN(C)C)NCC1CCC(C)O1)SC N1(C(C(Cc2n(C)cnn2)N)=O)CCC(S(=O)(=O)c2ccc(Br)cc2)CC1 N1(C(c2c(CC)ncnc2)=O)CC(NC(C2(OC)CCS(=O)(=O)C2)=O)CC1C N(C(=NCCCCl)NCC(C(F)(F)F)N1CCOCC1)Cc1cnc(C(C)C)o1.SCC N1(c2nc(C)nc(Cl)c2)CC(NC(=O)C2=C(Cl)CC2)C2CCCCC12 N1(C(c2cc(C(C)C)on2)=O)CCC(NC(=O)CC2CC(F)(F)C2)C(C(C)C)C1 c1(OC)cc(C(=O)NCc2ncccc2C(=O)N(C)C)ncn1.C(C)(CC(=O)OC)N N1(C(CCC(C)(C)NC(C(n2ccc(C)n2)C)=O)=O)Cc2cccc(F)c2C1 c1(C(=O)NC(c2ccc(C(F)(F)F)cc2)C(=O)OC)cc(C)cc(F)n1 C#Cc1ccc(C(=O)NC(C)CNC(C2(C)CC2C)=O)cn1 c1(CC(=O)NC2(CN3CCC(SC)CC3)CCC2)ccc(-n2cncn2)cc1 C1(C(=O)OC)CC2CCC1N2C(=O)C(O)C1CN(C(C)=O)C1 C1(C(=O)NCC(CC=C)CC=C)CN(C(c2cc(C)cc(C)n2)=O)CCC1(C)C N1(C(c2cc(C)on2)=O)CCN(C(=O)Cc2ccc(O)cc2Cl)CC1C(C)(C)C N1(CC)CCC2C1CCCN2C(=O)C(=O)N.c1(C=O)ccccc1 C1(C(=O)NCC2(C(N)=O)CN(c3ncc(C)cn3)C2)CC2(C1)NC(=O)NC2=O N1(C(C(C(=O)OC)(C)C)=O)CCC2(CCC(NC(c3n[nH]c(C4CC4)n3)=O)C2)C1 N1(C(CCN(CC#C)C(c2ccn(COC)n2)=O)=O)CCCC2(CC2)C1 N(C)(S(=O)(=O)N(C)C)CC(=O)NC1(CCO)CN(C(C=Cc2nc(C)sc2)=O)C1 C1(N(C(C(C(C)C)SC)=O)C)CCCCN(C(c2ccc(C)nc2O)=O)C1 C1(C(NOCC#C)=O)CCN(C(=O)CCC(C)SC)CCO1 c1(C(=O)NCC(=C)CCNC(=O)C(C)=CC(C)(C)C)ccc(Cl)c(F)c1 C12(C(=O)NCCCC(C)NC(COC(CC)(C)C)=O)CC1COC21CCC1 c1(NC=O)ccc(C(=O)NC2CN(C(c3cc[nH]n3)=O)CC2F)cc1 N(C1c2ccccc2CC1NC(=O)C=CC1CC1)C(c1ccc(C(N)=O)nc1)=O N1(C(CC2(OCC)CC2)=O)CC(O)CCC1C(=O)NC(c1nncn1C)CO c1(C(N(CCNC(C(C2CCC2)OCC)=O)C2CC2)=O)cc(I)c[nH]1 C(N=C(NCc1cccc(C(F)(F)F)c1)NC1CCCS1)C1(OC)CCOC1 N1(C(c2n(CCOC)ncc2)=O)CCC(C)(NC(c2cc(Br)ccc2F)=O)CC1 CS(=O)(=O)c1ccc(C(=O)NC2(CCNC(C3CC4C=CC3C4)=O)CC2)o1 N(C1CCCc2c1cnn2C)C(C1CCN(C(C(C(C)C)O)=O)C2C1OCC2)=O C12(NC(C(C)(C)O)=O)CC3CCC(C1C2)N3C(C1(C(=O)N)CC1)=O.C12CC(CC1)O2 CCCC(CCCNC(C1CC1Cl)=O)NC(=O)C=Cc1cncs1 c1(NC)cncc(C(N2CCC(CN(C)C(c3cc(C(F)(F)F)no3)=O)C2)=O)c1 N1(C(CSC)=O)CCC2(CCOC2)C(CNC(c2n[nH]c3cc(C)ccc23)=O)C1 CCC(Cc1ccccc1)CC(=O)Nc1cnnn1-c1ccc(Cl)nc1 CC1(CCO)CCN(C(c2cc(NCC3=CCSC3)ncn2)=O)C1 n1(CC)nc(C(C)C)cc1C(N1CCN(C(=O)COc2ccon2)CC1)=O CC(CC(=O)N1CC(C)(NC(C2CCN2C)=O)C1)C(F)F N1(C(c2c(CC)[nH]cc2)=O)CCCCCC1CNC(=O)CSc1cn(CC)nn1 C(C)(C)(C(C)CC(=O)NCc1noc(C(C)C)n1)NC(CC(CC)SC)=O C1(NC(C2CCCCO2)=O)CCC(C)(C)CC1.CC1C(=O)NCCC2(CC2)CO1 CCCCC(CCCC)NC(C1C(C)OCCN1C(c1ccnn1COC)=O)=O N1(C(CCCOCC=C)=O)CC2(CC2)CC1CNC(=O)C(C)(C)c1cnn(C)c1 C1(CC(N2CC(CNC(COCCOCC)=O)C(O)C2)=O)CCCC(C)(C)CC1 N1(C(C2=C(C)CC2)=O)CC(O)C(O)C1CNC(c1cccc(C(N)=O)n1)=O CN(S(N)(=O)=O)CC(N1CCCC1CCNC(c1cc(-c2ccns2)on1)=O)=O c1(C(=O)NC2CCN(C(C34OCC(C)(C3)C4)=O)CC2)ccc2c(c1)OCCO2 C1(CC)CN(C(=O)CCC[N+](=O)[O-])CCC1Nc1nccnc1C#N N12CC3C(C3C1)C2=O.n1(CC(=O)N(C)C)cc(CCC2CCCOC2)nn1 c1(C(CNS(NCC(=O)OCCOC)(=O)=O)OC)c(C)[nH]c2ccccc12 CCC(CC)CC(=O)N1CCCCC1CN(C)C(c1cnc(S)[nH]1)=O CC1CN(C(c2nn[nH]c2Cl)=O)C(C)CN1C(C1CC2CCC1CC2)=O C1(NC(C(n2cnc(C#N)n2)C)=O)CCC(F)(CNC(C2(C(F)F)CC2)=O)C1 CON1CC(C(N2CC(F)CC2CC(=O)NCC2CC3(CCO2)CC3)=O)CC1=O c1(Cn2cc(SCNC(CC3C(C)CCC3)=O)nn2)cccc2c1OCC(=O)N2 c1(C(N2CC(NC(C)=O)(CO)C2)=O)sc(C(C)=O)cc1Br S(=O)(=O)(CCC(F)(F)F)N1C2CN(S(CC#N)(=O)=O)C(C2)C1 N1(C(C(CCC)c2ccc(Cl)cc2)=O)CC2(CNC(=O)C=C(C)C)CC1CCO2 c1(C(=O)NC(CCNC(=O)C#CC2CC2)Cc2ccccc2)ccc(F)cc1Cl N1(C(C2CCCC2)CC)CCCCC1C1CCN(Cc2nccc(C)n2)CC1 C12(CCCSC1)NC2.S(=O)(=O)(CCN(C)C)N(CC)CC C1(OCCN(C(CN(C(COCCSC)=O)C)=O)C)CN(C)C2CCCC12 CC(F)CC(=O)NCC(Cc1ccccc1)N(C)C(c1csc(Cl)n1)=O CCCC(C)C(=O)NCC(C1CCCCCC1)NC(=O)CCC1CCCO1 CCC(C)(C)C(O)C(=O)N1CCOC(CCCNC(C2CC(O)C2)=O)C1 C1(CNC(=O)CC2(O)CCC2)CC2(CCN(C(c3coc(C4CC4)n3)=O)C2)CO1 c1(OC)ncc(C(=O)NC(C)CCCNC(c2coc(C(C)=O)c2)=O)c(C)n1 c1(C(=O)NCC2(NC(CC3CCCN(C)C3)=O)CCOC2)cc(F)c(Cl)cc1Cl c1(OC)cc(C(N2CCC(CNC(=O)C(C)C3CCCC3)C2)=O)nc(Br)c1 N1(C(C2N(C(c3ccn(C)c3)=O)CC(O)CC2)=O)CC2(CCCCC2)C1 N1(C(CCCN(C(C)=O)C)=O)CC(O)CC1C(=O)N(C)C(C1CCCC1)C N1(C(C(CC#C)NC(c2ccc(CC)cc2)=O)=O)CCN(CC)C(C)C1 CCC(C)C(=O)NCC(C(=O)N1CC(C(=O)OCC)C1)N(C)C N1(C(CCC(C)(C)F)=O)CCC2C(CCN2C(=O)CC2CCC(C)(C)O2)C1 S(=O)(=O)(c1cccnc1N(CC(C)C#N)C)N(CCCN(C)C)C C1(C(=O)NCCN(C(=O)C(C)(C)C2CCOC2)C)CC(=O)OC1(C)C C1(C(=O)Nc2cc(OCC)ncc2)CC(F)(F)CN1c1ncc(I)cn1 N1(C(C2N(C(C3N(C)C(=O)CC3)=O)CC=C2)=O)CC(F)(F)C(F)(F)C1 C1(C(N(C2CCCN(C(C3(C=C)CCC3)=O)C2)CC)=O)CCc2ccccc2C1 c1(NC2C(CC=C)CCCC2)cc(N2CCCC(F)(C(=O)NC)C2)nc(C)n1 CC1CCCn2c(CC(=O)NC3C4CC3N(C(C3CC3C(C)(F)F)=O)C4)cnc21 C1(CC)CCN(C(=O)CC2C(=O)NN=C2C)C(C(=O)N(CC(C)C)C)C1 C(=O)(CC(CNC(=O)CC(Cl)Cl)OC)NCC1(OC)CCC1 Cc1nn(C)c(Cl)c1C=CC(=O)NC(C)CN(C)C(C1CSCCS1)=O c1(C(N2CCC(N(C(C3CC(Cl)(Cl)C3)=O)CC)C2)=O)ccc2ccsc2c1 C#CC1(NC(C=C2CN(C(=O)CC3CSCCO3)C2)=O)CC(F)(F)C1 N1(CC(=O)Nc2cccc(OCC)c2)CCS(=O)(=O)CC1.C12(CC1)C(=O)NC2 N#Cc1c[nH]c2c(F)cc(F)cc2c1=NCC(O)COc1ccc(F)cc1 c1(OC)c(C(=O)N(C)CC2CCCN2C(C2CC23CCOCC3)=O)cccc1Cl C1(NC(C2CCC(=O)C2)=O)CC2CCC1CC2NC(c1ccncc1Cl)=O n1(COC)ncc(-c2nc(NC(=O)OC(C)(C)C)no2)c1COc1ccccc1 C(=O)(CCCC(=O)OCCSN1CCC(F)(NCC)CC1)OCC c1(C(N2CC(n3cc(CCCCC)nn3)C2)=O)cccc2nnn(C)c12 c1(C(=O)NC2CCCN(C(C(CCC)N(C)C)=O)C2)cc2c(cn1)CCCC2 C(=O)(C(C)C(O)C(C)C)N1C(CNC(c2ncc(OC)cn2)=O)CCC1 C1(C(C(=O)N(CC(C)NC(C2(CCC)CCC2)=O)C)C)CCOCC1 Cc1cc(N)c(C(N2CCCC(NC(=O)CC3CC3(Cl)Cl)C2C)=O)cc1C C1(NC(C2CC(OCC)C2)=O)CC(C)(NC(=O)C=C(C)C(F)F)C1 c1(OC)cncc(C(=O)NC2CC(N(C)C(c3ccc(C(N)=O)nc3)=O)C2)c1 Cc1ccc(C(=O)NC(CNC(=O)C(C)Oc2ccc(F)nc2)C(C)C)nc1 C1(CNC(C(C)(C)OCC)=O)CC(NC(=O)C=CCOCCOC)C1(C)C c1(OCC)ccc(C(C)=O)cc1NC(=O)C(N1CC(c2ccccc2)C(O)C1)=O N1(C(c2cnc(OC)c(Cl)c2)=O)CC(C)CN(C(C2(C#N)CCCC2)=O)CC1C C1(CNC(COCCN(C)C)=O)(CO)CCCN(C(C2CCCO2)=O)C1 C1(NC(C2C(NC)C2)=O)CCCCC1.c1(C(C(CCN)=O)=O)cnn(-c2ccccn2)c1 c1(N(CCCc2c(C)ccnc2)C)nc2c(c(=NC3CCN(C)C3C)[nH]1)SCC2 CC1CCC1C(=O)N(CCC(=O)N1CC(n2cnnc2)C1)C1CC1 CCCCCC(C)(C)C(=O)NCC(C)(O)CNC(c1c(C)[nH]c2ccccc12)=O c1(N(CCOCC)C)[nH]c(=NCc2cnc(C)cc2C)nc2sccc12 C1(CC(=O)N(CCNC(C(C2CCOCC2)C)=O)CCOCCO)CCS(=O)(=O)C1 C1(N(C(C2CCC(C)(CC)O2)=O)C)CCC2CN(C(c3ccc(F)s3)=O)CC12 C1(CC(=O)N(C2(CCN(C)C)CC2)C)CCCCCCC1.N12CCCC(C1)C2=O N#Cc1cc(C(F)F)cc(N2CCCC(Oc3ccccc3Cl)C2)n1 Cc1csc2ncnc(N3CCSCC3CNC(=O)CC34CCC(CC3)CC4)c12 CC1=NNC(=O)C1CCC(N1CCC(NC(=O)C(C)C(C)C)CC1)=O CCCCCC(CC)C(=O)N1CC(NC(c2ncsc2C)=O)CC12CCOC2 c1(C(=O)NC(CC)CN(C)C(c2cnnc(C)c2)=O)c[nH]c(=O)c2ccnn12 CC(C)(O)C#CC(=O)N1CCC(C(N2CCCC3(CCSCC3)C2)=O)O1 CS(=O)C=CC(=O)N(CCNC(C1CSCCS1)=O)Cc1cccc(Cl)c1 Cc1cc(C(N2CCC2CNC(C2CC(=C3CC3)C2)=O)=O)c(C)n1C N1(C(CCN(C)CC)=O)CC2(CCC2C(=O)NCCOc2cccc(OC)n2)C1 N1(C(C=CCCCCC)=O)CCC(C2(N(C(=O)CC3CC(OC)C3)CC)CC2)C1 C1(CCOC)(NC(=O)C(F)C(F)(F)F)CCN(C(c2coc(C(N)=O)c2)=O)CC1 c1(C(N(C2CCCNCC2)CCC2N(C)CCCC2)=O)ncc2ccsc2n1 c1(NC(C2CCC(NC(C(=O)OCC)=O)C2)=O)cccc2c([N+](=O)[O-])cccc12 c1(NC(=O)CN2C(=O)CSC2=S)nccc(I)c1C(N(C(COC)=O)C)C1CC1 N1(C(CCC=C)=O)CC(NC(=O)Cc2c(CC)noc2CC)C(F)(F)C1 c1(C(=O)NCCNC(C2C3CCC4C(C3)CC24)=O)cn2cccc(F)c2n1 Cc1ccc(CC(=O)N(CC(O)CNC(=O)Cc2ccc(F)cc2F)C)cc1F C(=O)(CC(C)(C)C(=O)N1CCN(C)C(CNC(=O)CSc2nc[nH]n2)C1)OC C1(NC(CNC(C2C(C)C2)=O)=O)CC=C(C(=O)N2CC(O)(C(N)=O)C2)C1 N1(C(COC)=O)CCN(c2cccc(F)c2)C(=O)C1.c12cnc(cn1)c(=O)[nH]2 C1(O)(CNC(C(C)N(CC)CC)=O)CCCN(C(c2cc(CO)on2)=O)CC1 N1(C(c2n(C)[nH]c(=N)c2)=O)CC(NC(C2CCCC(C(F)(F)F)C2)=O)CC1(C)C C=CC1(CO)CCN(C(C2CC(C)N2C(C2(OC)CCC(C)C2)=O)=O)CC1 c1(NC2(CNC(c3ccc(O)nc3Cl)=O)CCOCC2)ccc([N+](=O)[O-])c(O)n1 N1(C(c2cc(C)nn2C(F)F)=O)CCC2(CC2C(N2CCS(=O)(=O)CC2)=O)C1 CCCC(C(=O)NCC1CC(NC(=O)CC23CCC(CC2)C3)C1)NC(N)=O C(C(C)(C)C(=O)NC1CC(OCc2cncc(F)c2)C1)OCC c1(C(=O)NC2C3CN(C(CCC(=O)OCC)=O)C2C3)c(C)ccc2n[nH]cc12 CS(C)(=O)=NC(=O)C(=O)N1CC2CC2(CNC(C2CNC(=O)C2)=O)C1 CS(=O)(=O)C1(CN2CCC(CNC(=O)CC3C=CCC3)C2)CC1 CN1CCN(C(c2cc(=O)n(C)cn2)=O)CC1CNC(=O)Cn1cccnc1=O C1(NC(C2(CC#C)CC2)=O)CN(C(C2C3CN(C)CC23)=O)CCC1C N1(C(Cc2c(C)ncc(Cl)c2)=O)CCN(C(c2c[nH]c(C#N)c2)=O)C(C)C1C N1(C(=O)COCC2CCCC2)CCC2CN(C(c3ccc4[nH]ccc4n3)=O)C2C1 C1(CNC(C(N2CCOCC2)C)=O)CC2(CCN(c3cc(=O)n(C)c(O)n3)C2)CO1 CN1CC2(CCN(CCCCO)CC2)C1=O N1(C(CC(C)=C(C)C)=O)CCC(C(=O)NC(c2ccc(F)cn2)C)(CF)C1 c1(C(N(C2(CC(=O)N(C3CC(O)C3)C)CC2)C)=O)ccc(C#N)[nH]1 c1(CN)cc(C)ccc1N1CCCC1.C12CCCC(C1)NC(=O)NCC2 C1(C(=O)NCC(N(C(c2ncc(C)nc2)=O)C)C2CC2)CC2(CCCO2)C1 C1(C(=O)OC2CCCC2)CC(F)(F)C1.C1(C2CCC2)C(=O)NCCN1C c1(N(c2cncnc2)C)c(F)ccc(Br)c1F.c12cccc(c1)COCO2.OC N1(C(c2c(C)oc(CO)c2)=O)CCOC2(CCN(C(=O)C#CC3CCOC3)C2)C1 C1(CNC(C(C)(C)O)=O)C2CCC1CCN2C(c1sc([N+](=O)[O-])cc1Cl)=O N1(C(c2cnc(CC)nc2C)=O)CCC2CC1CN(C(=O)C(C)(C)C)C2 C1(NC(c2n(C(C)C)ccc2)=O)C2CCN(C(C3CCC(=O)N3)=O)CCC12 C1(NC(Cn2c(C(C)C)nnn2)=O)CN(C(=O)CCC2CCCC2)CC1(C)C C1(C(=O)NCc2cc(C(=O)NC(C3COCCO3)(C)C)n[nH]2)COCCN1C C(=O)(C(C)(C)CN(C)C(C1CCCN1C=O)=O)NCCC1CC(C)C1 CC(CF)CC(=O)N(C1CCCCC1NC(c1cnn(C(C)C)c1Cl)=O)C C(=O)(C1c2c[nH]nc2CN1C(=O)C(CO)OC)NCC#C c1(C(=O)NCCN(C)C(C2CC23CCOCC3)=O)cccc(Br)c1Cl c1(Sc2ccc(NC(=O)C(=O)NCC(F)F)cc2)nc2c(s1)CC(O)CC2 n1(CCOC)cc(C(=O)NCC(CC)(CC)NC(=O)C2=NOCC2)c(=O)cc1C c1(COC(CC2(C=C)CC2)=O)ccc2c(c1)OCO2.C123CC1CN(C2)C(=O)NC3 C(C)(CCCC(=O)N1CCN(C)CC1)NC(C1(CC=C)CC1)=O N1(C(C=CC)=O)CC2(C(=O)NCCN=[N+]=[N-])CC1CCO2 C(=O)(C(F)C(C)(F)F)N1CCC(C)(C(=O)NCCOC2CCOC2)C1 Cn1ncc(S(C)(=O)=NC(=O)C2CC3CC2C3)c1C(=O)O Cc1cnccc1C=CC(=O)NCC1C(C)CCN1C(c1nccc(Cl)c1O)=O c1(OC)c(Cl)cc(C(=O)NC2CC23CC(NC(c2c[nH]nc2C)=O)C3)nc1Cl Cc1ncc(C(N2CCC=CC2NC(CCOCCNC)=O)=O)cc1C#N C1(c2nnnn2C2CC2)(NCCN(C(C)=O)C(C)C)CCCCC1(C)C N1(C(c2ccc(C(C)(F)F)cc2)=O)CCN(C(C2CCCCS2)=O)C(C2CC2)C1 c1(OCC)ccc(CNC(C2CN(c3ccnc(C)n3)C2)=O)c(F)c1F C(=O)(CC(F)(F)CC(=O)N1CC2CC(C1)CN(C(=O)CNC(C)=O)C2)OC C1(CNC(=O)C(c2ccccc2)O)CC2(CO1)CN(C(=O)Cc1cc[nH]c1)C2 C(c1ccccc1)=C(OC)C(N1CC2CC1C2C(=O)NCc1nnc(C)n1C)=O c1(C(N2CC3C(C(=O)Nc4cc(OC)c(Br)cc4)(C3)C2)=O)cc(F)cc(C)c1O C(CCCCC(=O)Nc1cc(-c2ccccc2)no1)N(C)Cc1ccccc1.CCO Cc1ccccc1C(=O)N(C(C)CN(C(=O)Cc1cc[nH]c(=N)c1)C)C C(=O)(CC(C)(C)CC(F)F)N1CCC(C2(NC(CCC3N(C)CCC3)=O)CC2)C1 CC1(C)CCC(CNC(c2cc(Cl)c(Cl)[nH]2)=O)N(c2ncc(O)cn2)C1 c1(OC)ccccc1COC(=O)COc1ccc(CC2CN(C)CCO2)cc1 c1(C(=O)NCC2C(NC(CCCC(N)=O)=O)CCC2)coc2c1C(O)CCC2 CCC(C)CCCCC(=O)NCC1CC1C(=O)NCCc1ccnc(O)c1 O=C1Nc2ccncc2CC1OCc1cccc(C2CCCOC2)c1 N1(C(C2(CC)CCC(O)CC2)=O)CCC2(CCC2CNC(=O)C(O)C2CC2)CC1 C(CCC(C)C(=O)NCC(C(=O)N1CC(c2ccccc2)CC(C)C1)C(C)C)OC Cc1csc(C(N2CC(CNC(=O)C(=C3CCCCC3)F)C3CC23)=O)c1C C1(C(C)C)CCCCN1C(=O)C=CCN(C)C(c1ncn(C)n1)=O N1(C(CN(C)C)=O)CC2C=CC1C(C(=O)NOCC(C)(C)N(C)C)C2 N1(C(CCC=C=C)=O)CCC(NC(=O)COc2cncc(Cl)n2)C(CO)CC1 C(=O)(C1=CCc2ccccc21)NC1CC2CN(C(=O)OC(C)(C)C)CC(C1)C2 c1(C(=O)NC(CC(C)N(C2(C(=O)C(N)=O)CCC2)C2CC2)C)cccc(=O)n1C c1(CSCC)cn(CCN(C(=O)C(CC)N2CCCC2=O)C)nn1 N1(C(C(C(C)O)C)=O)CCN(C(c2nccc3cc[nH]c23)=O)C2(CCC2)C1 N1(C(C2CC(CCC)OCC2)=O)CCCN(c2ccccc2)CC1 C1(NC(CC2C(C)C2)=O)CC2CC(C1)N(C(c1cc(O)c(F)cc1N)=O)C2 Cc1cc(C(N2CC(N(C)C(C3CC4CCC3O4)=O)C(O)C2)=O)cc(N)c1Cl C1(NC(Cn2ccc(C)n2)=O)CC2CC(C1)N(C(=O)C=Cc1cnn(C)c1)C2 Cc1ncc(C=CC(N2CCC(C)C2CNC(=O)Cn2cc(C3CC3)nn2)=O)s1 c1(C(CNC(=O)C(C)SC(C)C)NC(c2c(CCC)n[nH]c2)=O)cccc(C)c1 c1(CCC(=O)NCC(CNC(C(C)=CC2CC2)=O)CO)ccccc1C#N C(=O)(CC(O)(c1ccccc1)C1CC1)NCC(C(C)C)NC(C1(C)CC1C)=O c1(OCC)ccc(C2(CNC(N3CCC(O)(CCC(C)(C)C)C3)=O)CCC2)cc1 CC1CN(Cc2cc(C3OCCO3)ccc2F)C(C)CO1.C1(=O)CO1 N1(C(c2ccc(CC)cc2F)=O)CCCC(C)(C)C1CNC(=O)CN1CCC1 N1(C(CCc2c(C)cccc2)=O)CCOC2(CCN(c3ccc(C#N)cn3)C2)C1 C1(NC(CNS(C)(=O)=O)=O)CC2CC1C1C2C1(F)F.C12CC(F)(F)CN1C2=O N1(C(CNC(c2ccc(C)s2)=O)=O)CCN(C(=O)CN2CC(C)C2)C(CF)C1 c1(C(N(CCNC(C2CCN(CC)C2)=O)CC)=O)cc2n(c1)CCC2 C1(C(N(C2CCN(C(c3nc(CCC)sc3)=O)C2)CCO)=O)CCC(=O)NC1 c1(C(=O)NC2CCN(C(C3C(COC)C3)=O)C(C)C2)ccc(C)c([N+](=O)[O-])c1 N1(C(C(CSCC)NC(=O)Cc2cn[nH]c2)=O)CCOC(C)(CC)C1 Cc1ccc(CNC(=O)Nc2ccnc(N3CCCCCC3)c2)nn1 C(C(O)C(=O)NCC(C)(C)NC(=O)OC(C)(C)C)=CCCC.C12CCC(C1)NC2 c1(CC(=O)N(CC(C)(C)NC(C2CC(C)(C)CCO2)=O)C)n[nH]c2ccccc12 c1(C(c2ccns2)NC(=O)NC23CC(C(F)(F)F)(C2)C3)cccc(F)c1 c1(NCC(CC)C(C)C)[nH]c(=NCC(C)(C)SCCO)nc2sccc12 C1(C(=O)NC2C(CNC(c3n(C)cnc3)=O)CC2)CC12CCOc1ccccc12 C#Cc1ccc(C(=O)NC(CC#CC)C(=O)N2CCCCC2CO)cc1C S(=O)(=O)(c1ccc(Cl)cc1)NCC(=O)NCCN1CC1=O.C(CC#N)S.CCCS.CC C(C)(C(C)(C)C(=O)NCC(CC)OC)NC(C=C(CCC)C)=O N1(C(COC(C)=O)=O)CCC(O)CC1C(=O)NCC1CCCCN1C C1(NC(C=CC(C)C)=O)CCCC(CC(=O)NCC2(F)CCOCC2)C1 C=C1CC(CC)C1.O1NC(=O)C2(CC2)N(C)C(=O)OCC(=O)NCC1 S(=O)(=O)(c1c(NC)ccc(Cl)c1F)NC.c12ccc(cc1)n(CC)c2=O C1(NC(C=COCC)=O)CCC2(CC1)CN(C(=O)C(CC(C)C)N(C)C)CCO2 c1(CCC(c2nnnn2CCF)NC(c2ncc(F)cc2F)C)c(Cl)cccc1Cl CC(F)(F)CC(=O)NCC1CCN1C(c1ccc(Nc2ccc(Cl)cc2)nc1)=O Cc1cc(C2CCC2)ccc1C(=O)NCCCC1CCCN1C(C1CC=CC1)=O Cc1c[nH]ccc1=NC(=O)C1CNC1.C1(N)CCCN(c2ncccn2)C1 C(CNC(n1nnc(C2CC2)n1)=O)(CC(F)(F)F)NC(Cc1c(C)n[nH]c1C)=O c1(C(=O)NC2C(C)CCN(C(C3CC(=O)C3)=O)C2C)cccc2c1nnn2C c1(CC(=O)NCCCOCCNC(C(C)C2CCC2)=O)ccc(C(N)=O)cc1 C1(C)(C(N(C)CCOCCCNC(=O)CC2CCCO2)=O)CC2C=CC1C2 C(=O)(C1CCCn2cncc21)NC(CC=C)CNC(c1cn(C)ccc1=O)=O c1(C(=O)NC(C)CNC(=O)C(C)(F)C(F)(F)F)cc2ccoc2cc1F CC(c1cnn(C)c1)=CC(=O)NC1CS(=O)(=O)CC1NC(c1cc(O)n(C)n1)=O c1(C(N2C(CNC(C3(C)CCCO3)=O)C=CC2)=O)ccc(S(N)(=O)=O)s1 c1(CCC(=O)NC2(C)CC(NC(c3ccc(C#C)o3)=O)C2)cnc2ncccn12 C1(NC(CCc2cc(OC)no2)=O)CN(C(C2(C)CNC(=O)C2)=O)CC(C)(C)C1 C1(N(C)C(C2CCC=CCCC2)=O)CCCN(CC(N2CCCC2)=O)CC1 Cc1sc(C(=O)Cc2csc(-c3ccc(C(C)C)cc3)n2)cc1CC(N)=O CCC(CC(=O)NC1CC(NC(=O)Cc2ccccc2C)C(O)C1)C1CC1 N1(C(C2(C#C)CCSC2)=O)CCC(n2cc(-c3ccncc3C)nn2)CC1 c1(C(=O)NCC(C)(C2CCC2)NC(C2Cc3nccn3C2)=O)cc2n(n1)CCC2 c1(C(=O)NC2CC3CN(C(c4cn(CC)nn4)=O)CC32)cnn2ccn(C)c12 CC(C(=O)N1CCN(C(=O)CCC2CCCCN2C)CC1)S(C)(=O)=O N1(C(C2N(C)CCN(C)C2)=O)CCC2C(CCCN2C(C2CC(CF)C2)=O)C1 c1(OC)ccc(C(CNC(C23CC(C2)C(C)O3)=O)NC(=O)CCC(C)C)cc1 C1(C(N2CCC(C(F)(F)CO)C2)=O)Cc2ccc(OCC(F)(F)F)cc2O1 O=C1C2Cc3ccccc3CN2C(=O)N1CC1(Br)CCOCC1 N1(C(CC2C(CC)C2)=O)CCOC2(CCC(NC(=O)C(C)(C)OC(C)C)CC2)C1 CC(=O)CCCC(C)C(=O)NC1CCCC(NC(C2CC(C)CCO2)=O)C1 C(C)(CCC(=O)NC1(CF)CN(C(=O)Cc2cccnc2Cl)C1)OC c1(C(N2CC3C(CNC(C(C)C4CC4)=O)C3C2)=O)cc(S(N)(=O)=O)co1 C1(CCCC)(C(=O)NC(CCN(C)C(c2cnns2)=O)c2cccs2)CCCC1 C1(NC(=O)OCCS(=O)(=O)NC(C)(C)C)C2CCC1(c1ccnn1C1CC1)C2 C12(NC(CNC=O)=O)CCC(C1)N(C(=O)CSc1nnnn1CC(F)(F)F)C2 C1(C(=O)NCCC2CN(C(=O)Cn3cnnc3)CCCO2)CCn2cnnc2C1 c1(C(=O)NC(COC)C(=O)NC(CO)CCCO)ccc(=O)n(C)c1 C1(N(C2(C(=O)NOCCCF)CCCC2)C(c2ccncc2)=O)CCCCCC1 C(=O)(CCCCN(C)C(c1cncn1C)=O)N(C)Cc1cc[nH]n1 Cc1ccc(SCC(=O)NCC2CCCN2C(c2cn[nH]c2)=O)cc1Br c1(C(=O)NCCOCCCNC(C(CCC)C)=O)cc2ccncc2s1 CC(F)(F)C(F)C(=O)NC1CC(COc2ccccc2)C1 Cc1ccc(C(=O)NCC(C)(F)CNC(=O)C(C)C)cc1F C12(NC(=O)Cc3cnns3)CCCCC1N(C(=O)CS(=O)(=O)C1CC1)CC2 c1(N2CCC(OCCNC(=O)CC(c3ccc(F)cc3)O)C2)ccnc2ncnn12 N1(C(c2c(C)n[nH]c2C)C(=O)NCc2nnn(C)n2)CCc2cccnc2C1 C(=O)(C(O)P(C)(C)=O)NCC1CC(OC)CN1C(c1cnn(C(C)C)c1C)=O c1(CN(CCCCCCCC)C=O)ccc2oc(O)nc2c1 C1(C(=O)NC(c2ccccc2)CO)CC12CCN(c1nnc(C(F)(F)F)s1)CC2 c1(OC)ccc(Cl)cc1C(N1CC2CC1CC2NC(c1cnc(F)c(C)c1)=O)=O C=CCC(CNC(C1CCCN1CC(C)C)=O)NC(c1cc(CO)[nH]n1)=O c1(NC(CSCCC)=O)cccc(NCc2cccc(-n3ccnc3)c2)c1 C1(CC)CN(C(C2(CF)CCC2)=O)CC1NC(=O)Nc1ncc(C2CC2)cn1 C(=O)(CCCCC(F)(F)F)NCC1C(C)(C)CCN(C(C2C(OC)C2)=O)C1 C1(C(N2CCC(C)C2(C)C)=O)CN(C(c2cc(C#N)ccc2N)=O)CC(C)(C)C1 C1(NC(CCCOCC=C)=O)CCC(C)N(C(=O)Cn2ccsc2=N)C1 C1(O)(CCNC(c2c(CC(C)C)onc2)=O)CCN(C(=O)C(O)C2CC2)C1 C1(CNC(C(C=C)O)=O)CC12CCN(C(=O)CCCCC#N)CC2 C1(C(=O)NCC2(F)CC(NC(CCC3(C)N=N3)=O)C2)CCC(F)(F)C1 Cc1ncnc(O)c1C(N1CCC(C(C)NC(C2(CO)CCCO2)=O)CC1)=O Nc1ccc(C(=O)NCC2CCC2NC(=O)CC(C2CCC2)C2CCC2)nc1 n1(CC)cc(Br)c(C(=O)NCC2CCN(C(=O)COc3ccc(OC)cc3)C2)n1 C1(C)(C(=O)NCC(N(C(CNC(CC)=O)=O)C)C2CC2)CCSCC1 c1(CC)cccc(OCC(N2CC(O)(CN(C(=O)CCC(C)OCC)C)C2)=O)c1 Cc1cc(C(=O)NCC(CC(F)(F)F)NC(=O)CC2CCCCN2C)cc(C)n1 N1(C(C(C)(C)CF)=O)CCC(C2(O)CC(NC(C3C=CCCC3)=O)C2)CC1 N1(C(C(CCCC)O)=O)CCN(C(=O)Cc2ccoc2)CC(C)(F)C1 c1(C2C(CC(=O)N(C(c3n(C)ccn3)C(F)F)C3CC3)C2)cccc(I)c1 c1(C(=O)N(C(C)(C)C)CCl)ccc(-c2cncnc2C(N2CCOCC2)=O)cc1F CC(C)CC(CNC(=O)CCc1ccc[nH]1)NC(=O)CC1CCN(C)C1 Cc1cc(Cl)n[nH]c1=NCC1CCCC1C.CC(C)CN C1(NC(c2c(COC)scc2)=O)CCN(C(=O)CC2CC3(CCC3)CO2)CC1F c1(C(N2CC(F)(CNC(c3c(C)nc(C(C)C)o3)=O)C2)=O)ncc2n1CCCC2 N1(CC)C(=O)CCC1CC(=O)N(C1CCN(C(c2cc(C)sn2)=O)CC1)C C1(NC(c2c(C)cnnc2)=O)CC2CCC1N2C(C1(C(F)F)CCCC1)=O N1(C(c2cn(CCC)nn2)C(=O)NCCC#N)CCC(C)(CO)C1 C1(CNC(c2c(C)oc(-c3cnn(C)c3)n2)=O)C(C2CC2)CCN1C(=O)C(F)F Cc1c(C(=O)N(c2nccc(Cl)c2F)C(C)C)ccc2cncn12 C(=O)(C(C)(C)CCC(C(=O)NCCC#N)N1CCOCCC1C(C)C)OCC c1(C(=O)NCC(C)NC(C(=O)NCC)=O)ccc(OCCF)cc1.OCC c1(C(C(=O)NCn2cc(SCC(N3CCC3C3CC3)=O)nn2)=O)ccc(F)cc1 C1(CCC(=O)NCC=C)CCCN(c2ncncc2C(F)(F)F)C1 c1(C(=O)NCCCNC(C(CO)NC(N)=O)=O)cc(N)c(F)cc1F c1(C(c2n(C(C)C)nnn2)NCCC2(CO)CC2)ccc(-n2ccnc2)c(F)c1 N1(C(c2nncn2C)C)CC2CN(C(c3ccc(-n4ccnc4)cc3)=O)CC2C1 c1(-n2c(C(=O)NCCn3cc(C(CSCC)C)nn3)cc(C)n2)ccc(Cl)c(Cl)c1 C1(CC(=O)NC(CC#C)CCOC)N(C(C2=NC=CS2=O)=O)CCC1(C)C c1(C(=O)NCCCN(C(C(=O)NC)=O)C2CC2)nc(Br)c[nH]1 N1(C(CCC)=O)CCC(C(=O)NCCN(C(=O)CC2CSC2)CC2CC2)CC1 c1(C(=O)NC(CC(C)NC(c2cn(CCO)nn2)=O)C)cccc2nnn(C)c12 CCCCCCC(F)C(=O)NC(CNC(=O)CS(=O)(=O)N1CCCCC1)CO Cc1c[nH]cc(C(N2CCC(N(C)C(C3CN(C4CCOC4)C3)=O)CC2)=O)c1=O C1(CC(N2CC(F)C(F)C2)=O)COCCN1C(C1CCCC(=O)C1)=O c1(N2CC(C(=O)Nc3cc(C)cc(O)c3)C(O)CC2)ncnc2cc(I)sc12 c1(CC)ncc(C(=O)NCC2CN(C(=O)CCC3CC3(Cl)Cl)CCO2)c(O)n1 c1(C(C)C(=O)NC2CCCC(C(F)(F)F)C2)cccc(-c2nn[nH]n2)c1 C1(CC(=O)NCC2(COC)CN(C(=O)CCc3nccn3C)C2)COC(C)(C)C1 c1(C(=O)NC(CCOC)CNC(=O)COCP(C)(C)=O)cc(=O)n(C)cn1 N1(C(c2cc(Br)n[nH]2)=O)C2CCC1CC(O)(c1ccccc1)C2 c1(CC)cc(C(N2CC3CC(NC(c4cc(OC)cs4)=O)C2C3)=O)cc(N)c1 O=C(CCCCC(F)(F)F)NCC(CO)NC(=O)CC1CC2(CCC2)CO1 C12(C(=O)NC3CCN(CC(=O)O)C(=O)C3)CCN(C1)S(=O)(=O)C2 N1(C(C(N2CCCCC2)C)=O)CCOC(C(=O)NC(C)CSC(F)F)CC1 c1(NC(C(N2CCC(F)(C(=O)OC)C2)=O)=O)ccc(F)cc1C(F)F C1(CN(C(=O)Cn2cccn2)C)CCN(C(=O)CCOCC(F)(F)F)CC1(F)F c1(CCC)ccccc1C(=O)NCCOCCCN(C(=O)C(F)C1CCOC1)C c1(N2CC(C)(CNC(Cc3n(C)cnc3)=O)OCC2)ncc([N+](=O)[O-])cc1CO N1(C(c2c(C)cnn2-c2ccccc2)=O)CCN(C)c2ccc(C)cc21 N1(CC2(C)CC2c2ccccc2)C(=O)CN(C)C1=O.CCC(C)(CN1CCCC1)OC C(CCN(C)C(c1ccc(CCC)[nH]1)=O)(C(C)C)NC(c1cn(CCC)nc1)=O N1(C(C(C(=O)OCC)F)=O)CCC(C)(C)C1CNC(=O)CC(=O)N(C)C C1(N(C)C(C2CC(C3CCC3)C2)=O)CCCCN(C(c2cccnn2)=O)C1 Cc1cc(C(N2CCC(NC(c3cc(N)cc(F)c3)=O)C2)=O)cc(C)c1F C1(NC(CC2N(C)CCC2)=O)CCC12CCN(C(c1cscn1)=O)CC2 CC1(C)CCN(C(=O)C#CC2CCC2)C1C(=O)NCc1ncc(F)cc1F c1(COC)ccoc1C(=O)NCCCC1CCCN1C(=O)C(O)c1ccsc1 c1(C(=O)NCC2N(C(CCCCOC(C)C)=O)CC2)cc(Cl)c2ccccc2n1 C12(CNC(C3C(C)(C)C3(F)F)=O)CCCC1N(C(c1coc(O)n1)=O)CC2 CC(C)CNC(=O)CN(C(=O)CNC(C1(Cl)CC1)=O)C C(=O)(CC(C)(C)CCOC)N1CC(N(C(c2c(CC)[nH]cc2)=O)C)C1 C(=O)(CC(=O)NN1C(CC(C)(C)Cn2cc(-c3ccns3)nn2)CCC1)NC.C1(C)CC1 N1(C(C(n2ccc(C)n2)C)=O)CC(O)CC1C(=O)NCC(C)(C)CC1CC1 C(C)(C(C(=O)NCCC1CCOC1)NC(c1cc(C)sc1N)=O)OC c1(C(N2CC(C(C)NC(=O)Cc3ccc(Cl)s3)C2)=O)cn2c(n1)CCCC2 c1(C(N2CCCC(N3CCN(C(CCC#C)=O)CC3=O)C2)=O)cc(F)cc(I)c1 N1(C(C2CN(C(CC)=O)C2)=O)CCCCC1C1CCN(CC2CCOC2)C1 C1(C(N2C(CC(=O)NC)CC2)=O)CN(C(=O)C(F)F)CCN1C C(=O)(CCCCCCNC(C1(OC)CC(C)(C)C1)=O)N1CC(C2CC2)(OC)C1 Cn1cnc(C=CC(=O)NCC2CCN2C(c2cc(-n3ccnc3)cs2)=O)c1 C1(CN(C(=O)C(Cl)=CCl)C)CC(F)CN1C(=O)CSCc1cccs1 CN1CC2CCC(C1)N2C(C1(C)C=CCN1C(C1CCC(C#N)CC1)=O)=O c1(OCC)ccc(=NC(=O)CCC2CCN(C(=O)C(C)(C)Br)CC2)[nH]n1 N1(C(C(n2cc(-c3cc(CO)ccn3)nn2)C)=O)CC2CCC(C1)C(=O)O2 C1(NC(c2csc(O)n2)=O)CC2(C1)CN(C(c1cnc(C(F)(F)F)cn1)=O)C2 c1(C(C(=O)NCC(F)=CC)NC(=O)OC(C)(C)C)ccc(F)c(Cl)c1.O=C(O)CO C1(CC(=O)N(CCC(=O)NCc2cnsc2)C)C(C)(C)CO1 c1(CNC(C(C)OC2CCCC2)=O)ccnc(C(N2CCNC(=O)C2)=O)c1 N1(CCNC(=O)C(O)CF)CCCN(C(c2ccn(-c3ccccc3)n2)=O)CC1 c1(OC)cc(C(F)(F)F)ccc1-c1cc(C(N2CC(CO)OCC2C)=O)ccn1 N1(C(CC(C)OC)=O)CCOC2(CCCN(C(=O)Cc3cc(Cl)cnc3C)C2)C1 C1(C(N(C2CCOC2)C)=O)(NC(=O)C=Cc2ccco2)CCSC1 Cc1cncc(C)c1C(N1CCC(C(=O)NC2CCCN(O)C2=O)C(C)C1)=O c1(OC)cc(F)c(C(N2CC(NC(C3CCC(C)(C)C3)=O)CC2(C)C)=O)cc1N c1(C(N2CC(=C(CNC(c3c(CC)non3)=O)F)C2)=O)cc(O)nc(O)n1 c1(CC(=O)O)ccc(-c2csc(C(N3CCCC3CC(=O)C(=O)O)O)n2)cc1 C1(C)(C(=O)NC(CN(C(=O)CSS(C)(=O)=O)CC)C)COCCO1 C(=O)(C1=NN(CC)C(=O)CC1)N1CCC(CNC(C(CC)C(F)(F)F)=O)C1 C12(CC(=O)NC3(CO)CN(C(=O)CC4CC5CCCC45)C3)CCCCC1C2(F)F C(C(N=[N+]=[N-])C(=O)NC1CCCCC1NC(c1ncccc1OC)=O)OCC C1(C(=O)NCC2(NC(C3NC(=O)OC3)=O)CCC2)CCC(C2CC2)C1 CC1CN(C(c2ccc(SC(F)F)cc2)=O)CC1NC(c1coc(O)n1)=O C(C#Cc1cn(C2C=CCCC2)nn1)NC(c1noc(C)c1C)=O C(=O)(CC(C(F)(F)F)NC(C1CN(C)CC(C)O1)=O)NC(CC)CCO CCC(C(=O)NC1(CNC(C2(C)CC2(C)C)=O)CCCCC1)C(C)C c1(C(=O)NC2CN(C(C(C)NC(N)=O)=O)CC2C)cc(O)nc(N(C)C)n1 C(=O)(CCF)NCCN(C(C1(C(=O)OC)CCC1)=O)CC Cn1c(=O)oc2ccc(C(=O)CN3CCCCC3CC(=O)O)cc12 N1(C(C2(N(C(c3nc(C)c(C)s3)=O)C)CC2)=O)CCCC2(CCC2)C1 C(=O)(C(C)CCCC(C)C)NCCCOCCCCNC(C(C)OCCCC)=O N1(C(C2(NC(c3nc(C)oc3)=O)CCCC2C)=O)CC(CO)C2(CCC2)C1 Cc1cccc(C)c1OCC(=O)N(CCCNC(c1ccsc1C)=O)CCOCF C1(C(N2CCC(n3cc(-c4ccnc(F)c4)nn3)C(O)C2)=O)CCC(F)(F)CC1 CCCCC(C(=O)NC)NC(=O)CNC(=O)CNC(C1CC1CCOC)=O N1(C(C(N)=O)=O)CCN(C(C2CC3CCC3C2)=O)CC1CF C(CCC(C)(F)F)N(C)C(C1CN(C(c2ccc(C(F)F)o2)=O)CCO1)=O N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(=O)C(C)(F)F)C(C)(C)C1 CC1CC(NC(c2ccsc2C(F)(F)F)=O)CN1C(c1cc(Br)no1)=O N1(c2snc(COC)n2)CCC(NC(C2CCCS(=O)(=O)C2)=O)C(O)C1 c1(-c2cn(CCCC)nc2)ccc2cc(C(=O)NC(C)CCO)cn2c1 N1(CC)CCOC(C(=O)NCC(C)(C2CC2)NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 CC1CN2CCN1CC2C(=O)N(CCCCCNC(=O)Cc1ccsc1Cl)C CC1(C)COC(CC(=O)NC2(CF)CCN(C(=O)CC3CCCCC3O)C2)C1 N1(C(c2n(CC)ccc2)=O)CCCC2(NC(C3CC(O)C3)=O)CCCC12 c1(C(N(C2CC2CNC(c2cccc(OCC(F)F)c2)=O)C)=O)ccc(N)c(N)n1 C1(NC(C2CN(CC)C(=O)C2)=O)CCN(C(=O)CCc2cccc(Cl)c2)C12CC2 c1(OC)cc(Cl)c(S(=O)(=O)N2CCc3ccc(C)cc3C2C)cc1Cl CC(C(=O)N1CC(N(C)CCNC(=O)C=CBr)C1)C1CCCC1 c1(-c2[nH]nc(C(=O)NCc3nc(CNC(C(N)=O)=O)sc3)n2)ccc(F)c(F)c1 C1(c2cn(CC3N(C(c4c(C#N)csc4)=O)CCC3)nn2)CCC(F)(F)CC1 c1(C(=O)NCC2(C(C)(C)O)CN(C(CN(C)C)=O)C2)ccc(F)c(O)c1 c1(C(=O)NCC(C(C)(C)C)NC(C(CC)n2cccn2)=O)cc2n(n1)CC1(CC1)C2 C(=O)(CC1=CCN(C(=O)CC(C)F)CC1)N1CCCC(C)(OC)C1 c1(C(=O)NC2(C)CC(NC(C3C(CC)OCC3)=O)C2)cc[n+]([O-])cc1 Fc1ccc(C(CCSC2CC3CC3C2)Oc2cccnc2)nc1 N1(C(Cc2c(C)noc2C)=O)CCN(C(=O)Cn2ccnn2)C2CC12 CC(C(C)C(=O)NC1(c2cn(CCN3CCCCC3)nn2)CCCC1)S(C)(=O)=O CCC(CNC(c1c(CNC(c2cc(C3CC3)[nH]n2)=O)nnn1C)=O)CCO C(CCCCC(=O)N1CC(C)OC(C)C1)N(C(CC(C)OC)=O)C c1(NC2CCN(C(C3(CC)CCC3)=O)C2)ncncc1C#N n1(CCN2CCN(c3nccc([N+](=O)[O-])c3)CC2)cnc2cc(Cl)ccc12 c1(CNC(C(C23CCC(CC2)C3)N(C)Cc2ccc(Br)o2)=O)ccc(F)cc1 CCC(C)C(C(C(=O)NCCC1CC1)N(C)Cc1cccc([N+](=O)[O-])c1)OC CC1=CCC(C(=O)N(CC(O)CN(C(=O)C(C)(C)c2ccsc2)C)C)CC1 Cc1nnccc1C(=O)NC(C1CCCC1)CNC(C1(C2(C)CC2)CC1)=O N1(C(CCc2cc(C)c(Cl)cc2)=O)CCC(C)N(C(C2CC2C)=O)CC1 C(=O)(C1=Cc2cccc(OC)c2OC1)Nc1ccc(NC(COC)=O)cc1C c1(OCC)cc(CNC2CNCC2CO)cc(Br)c1OC(F)F C1(NC(CN(C(C)C)C)=O)COCC1C(=O)N(C1CCOC1)CCO c1(CN2CC(CC)N(C(=O)C(C)(O)C(C)C)CC2)ccc([N+](=O)[O-])cc1F CCC(C)(CC)C(=O)N1CCN(C(c2cccc(OC)c2N)=O)C(CCOC)C1 c1(NC(N2CC3CCCC(C3)C2)=O)cnc2[nH]cnc2c1 C1(NC(C(C2CCN(C(C3CC3(C)C)=O)CC2)C)=O)CCOC(C)(C)C1 c1(C(N2CCC(C)(C(=O)Nc3cc(C)c(O)cn3)CC2)=O)ccc(O)c(F)c1F c1(CCC)ncc(C(=O)NCCCN(C(C2CCC(C(N)=O)C2)=O)C2CC2)s1 C1(N(C(=O)CCCn2cncn2)CC)CCN(C(=O)C(F)C2CCC2)CC1 Cc1ccc(C=CC(N2CC(C)(NC(c3cnccc3C)=O)C2)=O)s1 c1(CO)c(Cl)cccc1Cl.c12nc(cs1)CCNC2c1nnnn1CCCF C(=O)(CCC(CF)CF)NC(CC#C)(C)C(=O)NCc1ccc(Cl)o1 O=C(CC(F)(F)C(F)F)NC1CC1CNC(c1ccn(CCC(F)(F)F)n1)=O N1(C(CC=CCC)=O)CCC2CCC(NC(=O)CCNC(=O)CO)C1C2 C1(C(N2CC(CCO)(NC(=O)C3=CCCC3)C2)=O)Cc2c(F)cccc2O1 C(=O)(C(C)CCC(C)(C)C)NC1CC2(CC(C(=O)NCCNC(C(C)C)=O)C2)C1 N1(C(CC(C)OC)=O)CC2CCN(C(c3ccc(NS(C)(=O)=O)nc3)=O)C2C1 C1(C(N(CC)CC)=O)C(C)OCCN1C(=O)C=CCCC(C)C Cc1ccc2c(c1)CN(C)C2=O.c1(S)ccccc1F.c1(N)ccccc1 N1(C(C(=O)NCCCC=C)=O)C2CCC1CC(F)C2 C1(C(=O)NC(CNC(c2cc(C(F)(F)F)n[nH]2)=O)C2CC2)CCn2ncnc2C1 C1(C(=O)NCC2(C)CCCCC2)COCCN(C(C2OCC3CCCC23)=O)C1 C#Cc1cnc(N2CCC(CNC(c3cnc(F)c(F)c3)=O)C2(C)C)nc1 C1(C2CN(C(=O)CCCCC3CC3)C2)(NC(C2C(C)C2)=O)CC1 N1(C(C2C(C)=CCS2)=O)CCCN(C(c2cc3c(s2)CCC3)=O)C(C)C1 c1(N2C(C)(CNC(C3(C)CCCS3(=O)=O)=O)CCC2)nccn2nnnc12 N1(C(CC2CC(C)C2)=O)CCC(CO)(CNC(=O)C=Cc2ccc[nH]2)C1 c1(NC(=O)NC(C(=O)NC2C(C(=O)OCC)C2)C)c(Cl)cnn1C1CCCC1 N1(C(c2ncc(C)cc2C)=O)CC(C)(C)OC2(C1)CN(C(c1[nH]cnc1C)=O)C2 C(c1ccc(C)nc1)=CC(=O)N(CC(CC)NC(C1CCC=CCCC1)=O)CC Cc1ccc(F)c(C(N2CC(NC(C3CC(OC(C)(C)C)C3)=O)CC(O)C2)=O)n1 CCCCC(CNC(c1sccc1C#N)=O)NC(=O)CC1CC2CC2C1 CCC(CC(=O)NCc1ccncc1)NC(=O)C(C)CSC C1(CC(=O)NCC2(F)CN(C(C3CCCN3C3CC3)=O)C2)CCC(C(F)(F)F)CC1 Cc1ccn(C)c1NC(=O)CS.c1(CCC(=O)N(CCC(C)N)C)c(C)n[nH]c1C Cc1cc(C(=O)NC2CCN(C(c3nc(=O)n(C)[nH]3)=O)CC2CO)cc(C)c1Cl c1(C(=O)NCC2C=CC(NC(CNC(=O)OC)=O)C2)cc2scnc2[nH]1 Cc1nnn(CC(=O)NCC(c2ccccc2)N(C(=O)Cc2ccccn2)C)n1 C1(NC(C2CCC(CC)CC2)=O)CC1C1CCCN(C(c2ccc(C)n2C)=O)C1 N12CCC(F)(C1)C(=O)NC(=O)C1(CCC1)C2=O.N1(C(C)(C)C)CCC1CC1CC1 C12(NC(=O)Cc3ccc(CO)cc3)CCCC1CN(C(=O)C1=COCC1)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCC2CN(C(=O)Cc3cc(C)sc3C)C2C1 CCCCCCN(CC(N1CCC(NC(=O)CC2CCCSC2)C1)=O)CCSC C12(NC(CCOCCOC)=O)CCC(NC(C3CCCC3C(F)F)=O)(CC1)C2 C(CCN=c1[nH]c(=NCc2cccnc2N(C)C)[nH]c2ccsc12)OCC N1(C(C(c2cnccn2)C)=O)CC(NC(=O)C=CCSc2ccco2)CCC1C c1(C(N(CC(CNC(CCOCCC)=O)C)C)=O)ncc(OC)nc1OC c1(C(=O)NCC2N(C(C=C(C)C3CC3)=O)CCCC2)cc(Cl)ccc1C c1(C(N(CC)CC2CCCN(C(=O)CCCCCF)C2)=O)ccc(N)c(Cl)c1O N1(C(C(C(C)C)SCC)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)CC1CCO c1(C(=O)NC2CCCC(N(C(CCOCC#C)=O)C)C2)ccc([N+](=O)[O-])cn1 C1(OC)CN(C)C(C)(C(=O)NC2CCN(C(c3ncc(Cl)n3C)=O)CC2)C1 C1(NC(C23CC(CNC(C(C)(F)F)=O)(C2)C3)=O)CCN(C2CCC2)C1=O c1(C(=O)OC)cccc(CC(N2CCCC(NC(c3nc(O)c(C)s3)=O)C2)=O)c1 N1(C(Cc2c(C)noc2C)=O)CCC2(CCCN2C(C2CCC(C)(C)C2)=O)C1 c1(C(N2CC3N(C(C(CC)=O)=O)C3C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1Cl Cc1cc2[nH]c(C(N3CCCN(C(=O)CC(=O)NCC4CC4)C(C)C3)=O)cc2o1 c1(C(c2csc(Nc3ccccc3)n2)C(=O)NC)cc(Cl)ccc1OCCOC C1(c2cn(CCS(C)(=O)=O)nn2)CC(N(C(=O)C(O)CC2CCCC2)CC)C(O)C1 c1(OC)cc(N)c(C(=O)NCC2CC(NC(C3C(C)C3C)=O)C2)cc1S(C)(=O)=O N1(C(c2ccc(O)nc2)=O)CCN(C(c2ccccc2O)=O)C2CCCCC2C1 CC(C)C1=CCC(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])o3)=O)C23CC3)CC1 C1(NC(CSCCOC)=O)COCCN(C(c2ncsc2C2CC2)=O)C1 C1(C(=O)NCCN(C(=O)Cc2ccnc(O)c2)CC)CCC(C(C)C)CC1 c1(CC(=O)NC2CN(C(c3nc(C)sc3C)=O)CC2C)c[nH]c2c(F)cccc12 c1(C(=O)Nc2n(-c3c(CC)cccc3)ncc2C#N)cccc([N+](=O)[O-])c1Cl N1(C(c2n(CC=C)ccn2)=O)CCCC2(C1)CN(C(=O)C(=O)C(C)CC)CCO2 N1(CC)CCOCC1C(=O)NC1CN(C(=O)CC(F)(F)F)CC1C(N)=O N#CC1CCCC1NC(=O)CC1(NC(=O)CNc2c[nH]ccc2=O)CCCCC1 c1(OC)ccccc1C(O)C(=O)N(CC(C)Nc1cccc(NC(=O)CO)c1)C C(c1c(C)nn(C)c1Cl)=CC(=O)N(CCNC(CC1CC(C(C)C)OCC1)=O)C CCC(COC1CCCCC1)N=c1c(C#N)c[nH]c2ccc(Cl)cc12 N1(C(C(=O)NCCNC(C)=O)CC2(C)CC2)CCC(O)C(O)C1 C(=O)(CC1=CCN(C(C2CCCN2C(C)C)=O)CC1)NCC1N(C(C)=O)CCC1 c1(C(=O)NC(CC2CN(C(C(CC)C)=O)C2)C)cc(Br)c(Cl)s1 C1(C(=O)NCC(C2CCCC2)NC(C(C(C)C)(C)C)=O)CCCCN1S(N)(=O)=O N1(C(C2CN(C(CCCCOC)=O)CC23CC3)=O)CCC2(CCCC2)C1 c1(C(=O)NCC2N(C(C3(OC)CCCCC3)=O)CCC2C)cn2c(n1)SCC2 c1(-c2cc(C(=O)NC(C)(CCF)C(=O)O)on2)ccn2nccc2c1 C12(C(=O)NCC3CC(C)N(C(C4C(C)(C)C4(F)F)=O)C3)CCC(F)(CC1)CC2 N1(C(C=CC(CC)C)=O)CCCC(CNC(=O)C=Cc2cnc(C)s2)C1 C=C=C(C)CC(=O)NC(C)CN(C)C(c1cccc(OCc2ccccn2)c1)=O C1(c2nc(CC)[nH]n2)COCCN(C(C2C3CCCC23)C(=O)NC2CC2)C1 c1(OC)cc(NC(c2n[nH]cc2NC(c2ccc(Cl)c(Cl)c2)=O)=O)cc(Br)n1 Cc1cc(=NCc2ccc(CO)cc2F)[nH]c(NC2CC(O)C2n2cccn2)n1 Cc1nn(C)c(C)c1C(=O)NCC1CC(NC(C2CC(O)CN2C(N)=O)=O)C1 c1(OC)cnc(C(=O)N(C)CCNC(c2cnn(C)c2C)=O)c(OC)n1 CC(C)=C=CC(=O)N1CC(O)CC1CNC(C1CC2(CC2)CO1)=O CCC(CC)CC(=O)NC1(CNC(C2CC23CCCOC3)=O)CCCC1 Cc1cc(F)c([N+](=O)[O-])cc1C(N1CCOCC1CNC(=O)CCS(N)(=O)=O)=O Cc1cc(C(=O)N(C2CN(C(=O)C(C)(C)F)CC2F)C)c(S(N)(=O)=O)s1 N1(C(C2CCN(C(CC(CC(C)C)O)=O)C23CC3)=O)CCc2cccnc2C1 Cn1cc(NC(c2cn(CCOCC(=O)NOC3CCCCC3)nn2)=O)c(C#N)n1 C(CC(C)(C)C(=O)N1CCC(C)C(NC(=O)CC23COC(CF)(C2)C3)C1)OC Cc1nc(CNC(C2CC(C)N2C(c2nnsc2N)=O)=O)oc1C c1(C(N2CC(NC(=O)Cc3ccc(Cl)cc3Cl)C3C2C3)=O)cncc2[nH]ccc12 N1(C(C(CCC=C)NC(C23CC(CSC)(C2)C3)=O)=O)CCOC2COCC12 C#Cc1cc(C(=O)NC2(C)CCN(C(c3ccnn3C(F)F)=O)C2)cc(F)c1 C1(NC(Cn2nc(C)c(Cl)c2)=O)C2CC1N(C(=O)Cc1nc(C3CC3)cs1)C2C CC(C(=O)N1CCC(CNC(c2ncn3c2CCC3)=O)C(C)C1)P(C)(C)=O CC1CCCCN1C(C1CCN(C(=O)Nc2ccc(SCCC(C)C)cc2)C1)=O CCCC(C)(O)C(=O)N(CCCCCNC(=O)Cn1ccc(=O)cc1C)C c1(CC(C)C)ccc(C(=O)NC(C)C(C)NC(c2cc(Cl)c(Cl)s2)=O)cc1 C12CC3CCC(C1)N3C2=O.C=CC1CN(C(=O)Cn2ncccc2=O)CC1OC c1(CC(=O)NCC2(C)CC(NC(CCCOC)=O)C2)c[nH]ccc1=O N1(C(C2(C)C(C)CCCC2)=O)CC=C(CC(=O)NC2CC(CCF)C2)CC1 N1(C(c2cc(C3C(C)C3)no2)=O)CCC(c2cn(-c3ccncc3)nn2)C1(C)C Cc1cccc(C)c1NC(=O)C(c1ccc(F)cc1Br)N1CC(N(C)C)C(C)C1 c1(C(=O)CNC(CCC(F)(F)F)=O)scnc1C1CCCC1 CC(C)C(CCC(=O)N1CCCC(C(C)(C)C)C1)NC(c1ccn(C)n1)=O N1(C(CC(CC)CN(C)C)=O)CCC2(CCCN(C(c3ncccc3Cl)=O)C2)C1 N1(Cc2c(OC)nsc2)C2CCCC1CN(C(c1cncnc1)=O)C2 c1(C(N(C)CCOCCN(C)C(C2CC(F)C(=O)N2)=O)=O)cc(N)ccc1Cl c1(OC)c(F)cc(C(=O)NCCCN(C(=O)C(C)CSC)C)cc1Br c1(C(=O)NC(C)CCCNC(=O)C(F)=C2CCC2)ccc(C(F)F)cc1Cl c1(N(C)CCO)cn(CCNC(=O)OCCN2CCCC2=O)nn1 N1(C(c2ccccc2Cl)C(=O)Nc2ccc(OC)cc2)CC2OC(=O)N(C)C2C1 S(=O)(=O)(c1cccnc1NCc1cn(C)cn1)N1CCCC(CCC)CC1 N1(C(C2ON=C(C)C2)=O)CCC(C2(O)CN(C(=O)C3=C(C)CCOC3)C2)CC1 N1(C(C(C(=O)OC)C)=O)CCC2(CCCN(C(c3ccnc(Br)c3F)=O)C2)C1 CC(O)(CNC(=O)CC1CCCO1)CNC(C1(C(N)=O)CC1)=O CCCCC(CNC(C1CC1C(N)=O)=O)NC(c1oc(CCC)nc1C)=O c1(C(N2CC(CNC(C(COCC)(C)C)=O)OCC2)=O)cnc2n1CCOC2 C1(CC)CCCC(OCCO)C1.n12cc(nn1)CN(C)C(=O)CC2 c1(C(N(C2CCN(C(C(CC3CC3)OC)=O)CC2)C)=O)cc(O)nc(O)n1 C1(C(=O)NCC(C2CC2)NC(Cc2c(C)nc(C)s2)=O)CC(C)CC(C)(C)C1 N1(C(c2c(CC)ocn2)=O)C(C(=O)NC(C)CN(C)C2CC2)C2CC(O)C1C2 Cc1c(-c2nc(C(F)F)nn2C(C)C2CC2)[nH]c2cc(F)ccc12 C(N=c1cccc(C(C)=O)[nH]1)c1ncn(CC(=O)OC)n1 N1(C(CC2(OC)CCCC2)=O)CCCC(NC(C2CCCOC2)=O)CC1 N1(C(c2nn(CC)nc2Br)=O)CC2(CCCC2NC(=O)C=CC2CCOC2)C1 N1(C(C2(C)CCN(C(c3cccc(C=C)c3)=O)C2)=O)Cc2ccnn2CC1C N1(C(C(C(CC)C)OC)=O)CC2(C=C(C(=O)NCc3cnc(C)c(C)c3)CO2)C1 C1(C(N2CC(F)C2)=O)CCCC(F)C1.O=C1COCCN1 N1(C(c2nccc(NC(CCCOC(C)C)=O)c2)=O)CC2C(C1)C2(C)C c1(OC)ccc2c(c1)C(C(=O)N1CCC1n1cc(-c3cnc(C)n3C)nn1)CC2 C(CNC(c1ccc(CO)s1)=O)(CC(F)(F)F)NC(C(C)C1(O)CCC1)=O c1(CCC(=O)NCCN(CCOC)C(C2COCC(C)O2)=O)ccc(C)cc1C CC1CC(C)CN(S(=O)(=O)NC2Cc3nccn3C2)C1 c1(SC)ncc(Br)c(N2CCCC(C(N3CCC(N(C)C)C(F)C3)=O)CC2)n1 c1(C(N2CC(CNC(C=NOC)=O)C(O)C2)=O)ccc(OC)cc1O N1(C(c2n(C)cnc2)=O)CCC2(CC(NC(C3CCC3)=O)C2)C1 c1(C(=O)NC2CCN(C(c3c(C)c(Cl)ccc3)=O)CC2F)cc2cnccc2[nH]1 c1(N)ncoc1C1CCCO1.O=C(CCOC1CCC1)NCC(C1CCCC1)SC N1(C(Cc2cnc(C)s2)=O)CCC(NC(=O)Cn2nnc(=O)[nH]2)C(F)(F)CC1 CC(C)C(F)(F)CC(=O)NC1CCN(C(c2cn(Cc3ccccn3)nn2)=O)C1 c1(C(N2CC3C(NC(C(CC(C)C)F)=O)C3C2)=O)cccc2nccnc12 C1(CC)CN(C(c2ccc(C3CC3)cc2)=O)CCN1C(=O)C(CC)N(C)C CC1(NC(c2snnc2C2CC2)=O)CC(NC(=O)CCC2CC2(C)C)C1 N1(C(C(C)C(C)O)=O)CCC2(CCCN(C(=O)C(c3ccccc3F)(C)F)C2)C1 c1(OCCC(=O)NCCc2nc(-c3cccc(F)c3)no2)ccc(Br)cc1 c1(C(N(C2(CO)CCC2)C)=O)ccc(CNC(C2CC3CC3C2)=O)o1 C1(C(=O)NC(C(C)OC)C(=O)N2CCC(n3cncn3)C2)(CO)CC(C)(C)C1 C1(CNC(C2C(C(N(CC#C)C)=O)C2)=O)CCCCN(C(=O)CC(F)(F)F)C1 CCC(CCC(=O)NCc1cccc(CO)c1)OCCN(CC=CC(=O)NC)C Cc1cnc(N(CCC(C)C)CCC#N)c(S(=O)(=O)NC2CCS(=O)(=O)C(C)C2)c1 Cc1ccc(C)c(C2N(C(=O)NCC3CCCN3S(C)(=O)=O)C(C)C2O)c1.C(C)=O c1(OC)c(C)cc(C(=O)Nc2ccccc2CC2CCC3(CCC3)O2)cc1Cl N1(C(Cc2c(OC)nccc2)=O)CC(NC(=O)C=Cc2cscn2)C(C2CC2)C1 c1(C(N(C=O)CC2CN(C)C2)C2CC2)ccc(F)cc1 C1(N(C(=O)CCn2cccn2)CC)CCCN(C(c2ncccc2C)=O)C1 C=CC(CCC)CC(=O)N1CCC(NC(c2ccccc2N2CCCC2=O)=O)C1 C#Cc1ccc(C(N2CCOC(C(C)NC(=O)C(CCC)NC(N)=O)C2)=O)nc1 N(C1COc2cccc(F)c21)S(c1ccc(Nc2c(C)nc(C)s2)nc1)(=O)=O C1(CC)CN(C(c2csc3nccn23)=O)CCC1NC(=O)CC1(O)CCC1 CCCC(O)C(CO)NC(c1ccc(CC)cc1)CO N1(C(C2(SC)CCC2)=O)C2CN(C(C3CCC(C(F)(F)F)CC3)=O)CC12 c1(C(c2n(C(CC)C)nnn2)NCCCOC)scc(C)c1C(=O)ON(C)C N1(C(c2ccc(C#N)cc2Cl)=O)CCC2(CC1)CC(C(=O)Nc1nn[nH]n1)C2 C=CCC(CC(C)C)C(=O)N1CCCC1CN(C(=O)CC1CC(N(C)C)C1)C C1(C(=O)NCC23C(CN(C(C(C)Cc4cnn(C)c4)=O)C2)C3)CCC(F)(F)CC1 N1(C(CC)=O)CCCCC1C(=O)NC1CCN(C(c2ccn(C)c2)=O)C1CC C1(=O)C(C)(CC)Cc2nc1ccccc(NCCCCCC#C)[nH]2 Cn1ncc(C(=O)NC2CN(C(c3ccc(O)cc3)=O)C3CC23)c1Cl N1(C(CCS(C)(=O)=O)=O)CC2CCC(C1)N2C(c1ccc(F)cc1Br)=O n12cc(nn1)CC(C1CC1)C(=O)NCC2.C(C=CC(=O)O)(CC)=CC c1(C(N(C2CCCC(NC(Cc3c(C)scc3)=O)C2)C)=O)ccc(N)c(F)c1 C1(CNC(C(C)n2ccnc2)=O)CC2CC2N1C(=O)CN(c1ccccc1)C N1(c2nccc(C(=O)OCC)n2)CCS(=O)(=O)C(CCNC(=O)CSC(C)C)C1 c1(C(=O)NC(C2N(C(C(=O)NC(C)C)=O)CCC2)C)ccnc2c1nnn2C CCC(CNC(c1sc(NC2CC2)nc1C)=O)(CC)NC(C1CC(C)CO1)=O N1(C(=O)C2=CCOCC2)CC2CCC(NC(C3CC4CCC(C3)S4)=O)CC2C1 c1(CC)c(C(N2CCCC(CCNC(=O)C(O)C(F)F)C2)=O)cccc1C c1(C(=O)NCC(CNC(CC=CC=C)=O)C)cc2cccnc2s1 C(=O)(C(CC=C)CC=C)N(C1CCN(C(C2CC3(C2)CC3F)=O)C1)CC#C C1(CNC(c2cnccn2)=O)CCC(CNC(c2cc(C(F)(F)F)on2)=O)CC1 C1(C(N2CC3C(CNC(=O)CCc4ccccc4O)C3C2)=O)CC2(CCC2)CO1 Cc1n[nH]c(C)c1S(=O)(=O)NC1CN(c2ncnc3c(Br)csc23)C1 c1(C(=O)NCC2(C)CCC(NC(C(C)(C)C3CC3)=O)C2)c(F)ccc(N)c1F N1(CC(C)C)CCCC1C(N1CC(C(C)NC(=O)C=CSc2ccccc2)C1)=O c1(OC)ccc(NC(C2CCC(Nc3ncc(C(F)(F)F)cn3)CC2)=O)nc1Br c1(CN2CC(NC(c3cnc(C)[nH]3)=O)C(O)C2)cc(F)c(F)cc1O C(C(C)(C)CC(F)(F)F)NC(c1ccc(OCCCC)cc1)c1ccccn1 c1(C(=O)NCC2CCC(NC(C3(CC)CCC3)=O)C2)ccc(-c2cn[nH]c2)cc1 C1(C(=O)NC(CNC(c2cnn(C(C)(C)C)c2N)=O)CO)Cc2ccccc2C1 Cc1nc2c(n1C)CN(C(=O)Nc1ccc(OC(C)C)cc1)CC2 O=C(C1=CCOC1)NC1CN(C(c2cccc(-c3ccccc3)n2)=O)C2CC12 Cc1csc(=O)n1CCC(N1CCN(CC2CN(C(=O)C3CC3)C2)CC1)=O CC1=C(C(=O)NCC2CN(C(=O)C(C)CC3CCCO3)C(C)(C)C2)CCO1 c1(N(C)CCN2CCCCC2)ccc(-c2cc(CO)[nH]n2)cc1 C1(NC(c2ccc(C(F)F)cc2)=O)CN(C(=O)Cc2sc(O)nc2O)C2CC12 CC(C)C(C)(CNC(C1CC1F)=O)NC(c1cc[nH]c1)=O C1(C(=O)NC2CCN(CCOC)C2)(CC)CCN(C(=O)C=CC2CCC2)CC1 Cn1nc(Br)c2cc(NCc3nc4ccccc4[nH]3)ccc12 C1(OC)(CSC)CCN(C(c2ccc(C(F)F)s2)C(=O)NCC(C)C)C1.C1(O)CC1 c1(C(N(C(C)CNC(=O)CCN2CCCCC2)C)=O)cc(N)cc2ccccc12 C1(NC(Cn2ncc(C)c2)=O)CN(C(=O)C2=CCS(=O)(=O)C2)C2(CCOC2)C1 C=CCCC(=O)N1CCCC1C(C)(C)CNC(=O)Cc1cnccn1 c1(CC(=O)N(CCCNC(C2(C)CC(F)(F)C2)=O)CC)c[nH]c(=N)nc1O C1(NC(C=CC(C)(C)C)=O)CCN(C(=O)C=Cc2ccoc2)CCC1(F)F N1(C(CC2CC(=C)C2)=O)CCc2sccc2C1CNC(c1cn2c(n1)CCC2)=O Cc1cc(C(=O)NCCC(O)CNC(c2cnsn2)=O)cc(O)n1 N(C(=NCC1C(C)(C)C1(C)C)NCC1(C#N)CCOC1)C1C(C(C)C)C1 c1(C(C(=O)NC(CC)C)Nc2c(C(=O)OC)cccc2)nc(Cl)ccc1Cl CCN=c1nc(C(=O)NCC(C2CCOCC2)(C)OC)cc[nH]1 c1(OC)ccc(Cl)c(C(=O)N(C(C)CNC(c2csnc2C)=O)C)n1 C=CC(C)(CCOC)C(=O)N1CC(C(C(N)=O)NC(c2ccc3nccn3c2)=O)C1 c1(C(=O)NCCC(C)NC(c2cc[nH]c2-c2ccccc2)=O)ccc(F)cc1Cl C(=O)(CC1=Cc2ccccc2C1)NCC1CCN(C(C2C(C)(C(F)F)C2)=O)CC1 N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(=O)CCc2nccs2)C2CCCCC12 C(=O)(CC(CC(C)C)NC(c1ccc(C#N)s1)=O)N1CC(F)(C(=O)OC)C1 N1(C(c2c(CC)ncs2)=O)CC2CN(C(C3CCC3C)=O)CC2C1 N(C1CCCn2cnnc21)C(=O)CC1CCN(C(C2CC3CCCC3C2)=O)CC1 c1(C(N(C2CCN(C)CC2)CCCC)=O)ccc(S(N)(=O)=O)cc1Cl C=CCCC(CC(C)C)C(=O)N1CCCN(C(c2ccc(C(N)=O)s2)=O)C(C)C1 C(CCCC(=O)NC(C)CCF)NC(C(C)C1CCOC1)=O C(=O)(CC(C(F)(F)F)NC(c1ccc(F)c(C2CC2)c1)=O)OC C1(COC)(NC(c2cnn(C)n2)=O)CN(C(=O)CCc2ccc(C)o2)C1 c1(C(=O)NC2COCCN(C(c3nccc(C#N)c3)=O)C2)ccc2cnnn2c1 C1(CNC(c2cc(C)ncn2)=O)N(C(=O)CN2CCCC2C)CCC1(C)C N1(C(C(c2ccccc2)OC)=O)CCC(C2CC(NC(c3cc(C)c[nH]3)=O)C2)C1 C12(C(=O)NCCN(C(C(C)NC(=O)NC)=O)C(C)C)CCCCC1NC(=O)C2 C1(C(N2CC(C)(NC(c3coc(O)n3)=O)C2)=O)COCCN1S(C)(=O)=O c1(OC)cc(C(N2CCS(=O)(=O)CC2C2CC2)=O)c2cc(OC)[nH]c2c1 Cc1cccc2cc(C(=O)NCC3CN(c4cncc(Cl)n4)CCC3(F)F)[nH]c12 N1(C(CN(C(C)=O)C)=O)CCN(C(=O)Cn2ccc(O)nc2=O)C2COCC12 N1(C(CC2CCC(OC)CC2)=O)CCC(C)(NC(C2CCC=CCCC2)=O)CC1 O=C(Cc1cc2ccccc2s1)NNC(=O)N=c1cc2n([nH]1)CCCC2 CCC(O)C(C)C(=O)NCC1(O)CCN(C(c2cnc(C(C)=O)s2)=O)C1 N1(C(C=CC(C)C)=O)CC(CNC(C2(C)CCCS2(=O)=O)=O)C2(CC2)C1 C(N=c1[nH]c(N2CCC3(C2)CN(C)C3)nc(=N)[nH]1)C1CCC(C)(CC)O1 N1(C(c2ncccc2Cl)=O)CCC2C(C1)CN2C(=O)CCSCc1ccccn1 C(CN=C(NCc1cccnc1C)N1CCC(Cc2cnn(C)c2)C1)SC c1(CC)cnc(Cl)[nH]c1=NCCC1CCCN(C(=O)C2=C(Cl)CC2)C1 C(CC(C(=O)NCC1(CN=[N+]=[N-])CC1)NC(C12CC(F)(C1)C2)=O)N(C)C c1(NC(C2C3(CN(C(c4cc(OC)c(I)cc4)=O)C3)C2)=O)ccc2c(c1)OCC2 c1(C(=O)NC(C)CNC(=O)CC2(CS(C)(=O)=O)CC2)cnc(O)cc1C(F)(F)F C(C)(C)(C(C)CC(=O)NCC1CCC(F)(F)C1)NC(C1(C(C)(C)OC)CC1)=O CC(=O)CCCCC(=O)N1CC2CC1C2NC(c1csc(C)c1)=O N1(C(C(CCOCC)NC(=O)CC2C(=O)NN=C2C)=O)CC2(CC=CC2)C1 C1(CNC(C2C(CC)C2)=O)C(C)CCN1C(=O)CCN1CCNC(=O)C1 Nc1cccnc1C(N1CCCC1C(=O)NCCn1ccc(=O)cc1)=O c1(C(CNC(C(CC)C)=O)NC(=O)Cc2cccc(Cl)c2)ccc(F)cc1 C(=O)(C(F)(F)CO)N1C2CC(C2)C1.c1(C(=O)O)cnc(-c2ncccn2)s1 CCCS(=O)(=O)C(C)C(=O)NC1CCC(NC(c2cncc(C3CC3)c2)=O)C1 C(=O)(CCCC(=O)NC1(C)CC(NC(=O)CC(O)CC)C1)OCC C(C(F)(F)CNC(=O)C(C)(C)c1csc(=N)[nH]1)OC C12(CNC(CCC)=O)COCCN1C(=O)CN(C(c1cccc(CO)c1C)=O)C2 C(=O)(C(Cc1cccnn1)NC(c1ccsn1)=O)OC C(=O)(CC(C)(O)CCC)N1C(C(NOCCC)=O)CCC1 c12ccc(c3c1OCC3)[nH]c2=O.c1(C(=O)NCC)ncoc1C1CCCCC1 C1(C(=O)NCC(=Cc2ccco2)C)CCN(C(=O)C(C)=CC(C)(C)C)O1 CCCC(O)CC(=O)NCC(c1ccc(C)cc1)NC(=O)C(F)(F)C(O)C1CC1 N1(C(C=CCN(C(CC(C)c2ccco2)=O)C)=O)CC(O)C(O)C1 Cc1n[nH]cc1CCNC(C1(NC(c2csnn2)=O)CC1(C)C)=O c1(N(C)CC2CC2)nc(N2CCS(=O)C3(CCC3)C2)nc2c1CCCCCC2 C1(C(N(C)CCC2CCCN2C)=O)CC2CC2N1C(C1CCN(C)CC1)=O C12(C(=O)NC(C)C(CO)NC(=O)C(C)OC3CCCCC3)CCC(CC1)CC2 c1(CC)c(C(=O)NC2CCCC2CNC(=O)C(C)C(C)(C)C)cccc1F Cc1nc(C(=O)NCC2CCCCCN2C(=O)CC2CCCCC2)cn(C)c1=O N1(C(C(CC=C)NC(C)=O)=O)CCC2(CC1)CC2C(=O)N(CCCF)C N1(C(C2(C)CN(C)C(=O)C2)=O)CCN(C(C2CC(F)(F)C2)=O)CC12CC2 C=CCC1(C)C(=O)N2CCC(C2)CN1.C12CC1NC2=O.C(C)(C)(C)OC(=O)NC CCC(C)(C)C(O)C(=O)NCC(CC1CC1)C(=O)N1CC(C(F)(F)F)C1 C1(C(=O)NCC2C(NC(=O)CCc3ccsc3)CC2)CCC2CC2CC1 c1(C(N(CC(CN(C(C(C)NC(=O)NC)=O)C)O)C)=O)ccnn1C(C)(C)C Cn1cc2c(C(=O)NCC3CCN(c4ncnc5c4CCC5)C3)cccc2n1 N1(C(C2(COC)CCCC2)=O)CCC2C(C1)CN2C(c1cccc2scnc12)=O C1(NC(Cc2scc(C)c2)=O)CN(C(c2ccc(C(C)C)c(F)c2)=O)CCC1C C1(C(=O)NCC(CC=C)NC(=O)CCc2cc[nH]n2)CC2C=CC1CCC2 Cc1ccc2occ(C(=O)NCC34CC3CN(C(c3ccc(Cl)cc3)=O)C4)c2c1 CN1CC(O)CC1(C)C(N1CCCC(F)(C(=O)NCC2COCC2(C)C)C1)=O C1(C(=O)NCC(CC2CC2)CO)CN(C(=O)Cc2cc[nH]n2)CC1F C1(NC(Cc2c(C)cccc2C)=O)CC2CC(C1)N(C(C1CC(N(C)C)C1)=O)C2 N1(C(C2C3N(C(C4(C(C)(C)O)CC4)=O)CC(C=C3)C2)=O)CCN2C(=O)NCC2C1 c1(-c2c(OC)ccc(O)c2)cnc(C#N)c(C(N2CCC(CO)C2)=O)c1 C1(C(C)=O)CC(C(=O)NC2CC(NC(=O)C(F)(F)C3(O)CCC3)C2)C1(C)C C1(O)(CN(C(COC)=O)C)CCCN(C(C2CCC(=O)N(C3CC3)C2)=O)C1 CCC(CCC(=O)Nc1cccc(-c2c(C(=O)NC)cnn2C)c1C)OC.C(F)(F)F c1(CC(N2CC(F)CC(NC(c3n[nH]cc3Cl)=O)C2)=O)coc2ccc(F)cc12 N1(C(c2ccn(C)c2-c2cccc(Br)c2F)=O)CCC(F)(COC)CC1 N1(C(C2CCC(C)O2)=O)CCCC2CN(C(c3scnc3-c3cccs3)=O)CC12 CC1CC2(CCN(C(=O)C3=COCCC3)CC2)CN1C(C1CCCC(C#N)C1)=O c1(OC)ccc(-n2cc(CN(O)C(=O)CSC3CCC3=O)nn2)cn1 c1(CC)cn2c(n1)CC(C(=O)NCC1CCC(F)(F)C1O)CC2 C1(CCC)CCCC1C(N1CC(CNC(c2cnn(C)n2)=O)C2CC12)=O C1(C#N)(C(N2CCC(Oc3cc(OC)ncc3)C2)C(=O)NC(C)C)CCOCC1 C1(NC(C(CCCC)=O)=O)CN(C(c2cn(C(F)F)cn2)=O)C2(CCC2)C1 C1(N(CC(=O)Nc2nccn2C)CCC)CC2CCC1(C(=O)O)C2 O=C(C1=C(c2cc(F)ccc2)CCOC1)NC1CCCCCC1C(F)(F)F C1(C(N2CC(NC(C(C)(C3CC3)OC)=O)C(SC)C2)=O)CCC(C)(F)CC1 c1(C(=O)NCC2(O)CN(C(c3ccc(C)c(F)c3)=O)C2)cc(C)n(C)c(=O)c1 CN1N=C(C(=O)NC2CC(NC(c3cnc(Cl)cc3Cl)=O)C23CCC3)CCC1=O CC1(CCNC(C2(c3ccccc3)CCC2)=O)CCN(C(=O)CCF)C1 C(C)(CCC(=O)N1CCOC(CNC(c2cn(CCC(C)C)nn2)=O)C1)OC N1(C(CC(C)=O)C)c2ccccc2CC1C1(C(=O)O)CC1 c1(CNC(c2cccnc2O)=O)cc(O)nc(CNC(C2(CCF)CCC2)=O)n1 c1(OC)ccc(C(=O)NC(C)CC2CCN(C(c3cccs3)=O)CC2)c(C)n1 N1(C(c2nc(C)oc2)=O)CCC(NC(=O)C(c2cnn(C)c2)=O)CC1C c1(OCCC(=O)NCCN(C(C2CCN(C)C2)=O)CC)ccccc1C(C)C C1(C(N2C(CNC(CCN(C)CCO)=O)CCCCC2)=O)CCc2nccn2C1 C1(NCCC2(C)N=N2)CN(C(=O)OC(C)(C)C)CC12CCC2 CN1CCCCC(n2cc(CN(O)C(C3COC4CCCCC34)=O)nn2)C1=O C12(C(N3C(CN(C)C)CC(F)C3)=O)CCCN(CCC1)C2 N1(c2snc(CCC)n2)CCC(C)C(NC(=O)C(C)(c2ccccc2)N(C)C)C1 Cc1csc(C=CC(=O)NC23CC2CN(C(C2(c4cccc(Cl)n4)CC2)=O)C3)n1 N(C(=NCCCCS(C)(=O)=O)N1CCC(C(CN(C)C)OC)CC1)CC=C c1(C2C(C(=O)NC(CC)CNC(=O)Cc3nnc(C)o3)C2)cccc(C(C)C)c1 C(=O)(C1CCCc2ncnn21)NC1(C)CCCN(C(CCC#C)=O)C1 c1(-c2cn(-c3ccc(NC(C4CCN(C)C4)=O)cc3)nn2)cc2ccccc2o1 CCCC(C#N)C(=O)N1CC(NC(c2cc(-c3cnn(C)c3)on2)=O)CC1(C)C N1(C(COCC#C)=O)CC(N(C(=O)CC(CC)C2CCC2)C)C(O)C1 N1(C(C=CC=CC)=O)CC2CCC1C(CNC(=O)C(F)CC1CC1)C2 N1(CC(N2CCN(C(=O)C=Cc3ccc[nH]3)CC2)=O)CCc2cc(F)ccc21 c1(OC)ccc(C(=O)NCC2CC(OC)CN2C(C2CNC(=O)N2C)=O)cc1F c1(CNCC(=O)n2oc(=O)[nH]2)ccc(Cl)cc1.C1(Cc2ncc[nH]2)CCOCC1 CC1(C)CCC(C(=O)NC2(C(=O)Nc3cc(F)ccc3O)CCSC2)CO1 N1(C(CN(C)C(N)=O)=O)CCCC12CCN(C(c1cc(N)c(Cl)cn1)=O)C2 N1(C(C(CC(C)(C)NC(C2CC2C(C)(C)C)=O)F)=O)CCC12CCC(O)CC2 Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(=O)CC=C(Cl)Cl)C(C)C1 C(C)(c1ccccc1C)=CC(N1C(CNC(C2(CCC)CCNC2=O)=O)CC1)=O CC1(C)COC(CCNC(C2(NC(=O)C(F)F)CCCC2)=O)C1 C(=O)(C(COC)C(F)(F)F)NCC(C1CCCCC1)(C)NC(C)=O Cc1cccnc1C=CC(=O)NCCCN1CCN(C(C2(C)C=CCC2)=O)CC1 N1(C(CNC(c2n(CC)ncc2)=O)C(F)F)CCN(C(=O)CC2(F)CCC2)CC1 c1(OC)cc(N2CC3CC(NC(c4csnn4)=O)CC2C3)ccc1[N+](=O)[O-] C1(CNC(c2ccc(CC)cc2)=O)CN(CCOc2ccccc2Cl)CCCO1 C1(COC)CN(C(c2ccnn2-c2nccs2)=O)CCN1C(C1C=CCC1)=O CC(O)C(C)(C)C(=O)NC1CN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 NS(=O)(=O)c1ccc(C(=O)NC2CCC2NC(=O)Cc2ccoc2)c(F)c1 C1(O)(CC(N2CCC(Cn3cc(CN4CCCCC4)nn3)CC2)=O)CCCOC1 N1(C(c2n(C=C)nnc2)=O)CC(NC(C)=O)CC1(C)C C(c1ccc(F)c(Cl)c1)=CC(=O)NC1CC(NC(c2cccc(Br)c2)=O)C1 C(C)(C)(CC(=O)NC(C1CC2CCC1C2)C)NC(C(C)C1CC1)=O N(C(=NCCn1cccn1)NCc1ccc(C(N)=O)cc1)CC(C)(C)c1cccs1 C(=O)(CCC(=O)N1CCC(O)CC1)NCC(O)Cn1cc(CCSCC)nn1 N1(C(C2C3CN(C(C(C)Sc4cccc(C)c4)=O)C2C3)=O)CCCC2(COC2)C1 N1(C(c2c(C)nns2)=O)CCN(C(=O)C=Cc2ccc(F)cc2)CC1C(F)(F)F C1(CC(=O)NCC2(NC(CCC=CC)=O)CC2)CCCC(OC)C1 C(=O)(CCC(C)(C)C)NC1C(CNC(C2CCCN(C(C)=O)C2)=O)C1 N1(C(Cc2scc(C)c2)=O)CC2CCC(NC(c3ncnn3C(C)C)=O)CC2C1 C12(CC(n3cc(C4CN(C(=O)Cn5ncnn5)CCO4)nn3)C)CCC(CC1)C2 c1(C(=O)NC(C(=O)NCCCC(=C)C)CC(F)F)cc(C#N)ccc1N c1(OC)nscc1C(=O)NC1CC(O)C1CC(=O)NCc1nc(C2CC2)no1 C1(NC(c2cn(CCC(C)C)nn2)=O)CCN(C(=O)CCc2c[nH]c(=N)[nH]2)C(C)C1 CCC(CC)(CCC(=O)NC1C=CCN(C(=O)CC2(N(C)C)CCC2)C1)[N+](=O)[O-] C(=O)(C(O)C(F)(F)F)NCC(C)(C)CNC(C1(c2ccccc2)CCCO1)=O c1(C(=O)NC(C2CCCCN2C(=O)COC(F)F)C)ccc(N(C)C)cc1Cl c1(CC)nc(C)c(C(N2CC(C)(NC(=O)C(COC(C)C)NC(C)=O)C2)=O)s1 N1(C(C(C2CC2)OC)=O)CC(C2CN(C(c3ncc(Cl)cc3Cl)=O)C2)C1 CCC(C)(CNC(=O)C(F)(F)c1cccnc1)NC(c1cscc1Cl)=O C1(CC(=O)NCC2(C)CCN(C(c3c(C)ccnn3)=O)C2)CCC2CC1C2(C)C Cc1ccnc(C(=O)NC2CN(C(=O)Cc3nnn(C(C)(C)C)n3)C2)n1 CC1(C)CCOC1C(=O)NCC1(C)CCN(C(=O)CCCN2C(=O)CCC2=O)C1 CCCCC(CC)C(=O)N1CCC(C2CCCCN2C(c2cc3n(n2)CCO3)=O)C1 O=C1COc2cc(F)c(C(N3CCC(NC(C4CNC(=O)N4)=O)C3)=O)cc2N1 C1(C(=O)NC2C(CNC(CN(C)CC)=O)C2)CCCN1C1CCCC1 C1(CNC(c2c(C)nc(C(C)C)o2)=O)CN(C(c2cc(N)ccn2)=O)CC12CC2 c1(CN(C2CCC3(CC3)C2)C=O)ccc(F)c(C(F)(F)F)c1 c1(OC)c(C(N2CCC(CCNC(c3ccnnc3)=O)CC2C)=O)ccnc1Cl c1(C(N2C(CNC(=O)C3=CCCC3)CC3(CC3)C2)=O)cnc2[nH]ccnc1-2 O=[N+]([O-])c1cnn(CCN2CCOC(c3cn(CC(O)CO)nn3)C2)c1 c1(-c2nc(C)sc2)n[nH]c2c1CN(C(c1c(F)cc(O)cc1F)=O)CC2 c1(OC)ccc2ncc(C(=O)NC3COCC3CNC(=O)CO)n2n1 N1(C(C(CCC)C(C)C)=O)CCCC2CN(CCOc3ccccc3C)CCC12 c12ccnc(c1)CNC2=O.C12(CC)CCC(CO1)C2.c12cc(no1)C(C)NC2=O Cc1cc(C(N2CCC2C(=O)NC2CCCOC2)=O)c(C)cc1Cl CCC(C)(COC)CNC(=O)C(c1cn(C)nn1)NC(=O)C=CC1CC1 C(=O)(C1CCc2cccnc21)N1CC2(C(NC(C(C)=C(C)C)=O)CCS2)C1 C1(C(=O)NCC(C)(C2CCC2)NC(=O)CC23CC(C2)C3)CC2(C1)CC(F)(F)C2 N1(C(c2nnn(CC)c2C)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC1CF C1(C)(C(=O)NCC2(NC(Cc3c(OC)nccc3)=O)CC2)CCCC1(F)F C(=O)(C(C)Cc1ccncc1)NC1C(NC(CCOCCC)=O)CC1 CC1CCC(C(F)(F)F)CN1C(=O)NC1(CCO)CCCCC1 CCCC(C)CC(=O)NCC(C)OCC(=O)NCCn1cc(C)cn1 c1(C(N(C)CC2(CNC(CC(C)C)=O)CC2)=O)cnn2c(=O)cc[nH]c12 C(C(C(C)(C)C)NC(c1cc[nH]n1)=O)NC(C(n1ccc(C(F)(F)F)n1)C)=O C(C)(C)(CCCF)N.C1(C(N)=O)COCC1C(=O)NC.C12(CCCC1)C(=O)N2 C1(CNC(C(n2ccc(C)n2)C)=O)CC2(CCC2)CN1C(=O)OC(C)(C)C N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(CNC(=O)CCc2ccnc(Cl)c2)C1 C1(NC(=O)C=CCBr)CC12CCN(C(=O)Cc1ccc(F)cn1)CC2 c1(CC)ccc(C(=O)NC(C)CN(C)C(c2cc(CC)n(C)c2C)=O)cc1F c1(CC)ccoc1C(=O)NC(CC1CCCC1)C(=O)NC1CCCSC1 c1(CC)ccc(NC(=O)C(C2CCS(=O)(=O)C2)Nc2cccc(OC)c2)cc1Cl C1(C(N2CCC(CF)CC2)C(=O)NC(C)C)CCC2(CC2)C1 CC1(C)CN(C(C2(NCc3coc(Cl)c3)CC2)=O)CCO1.C(N)(=O)N N1(C(c2c(CC)cco2)=O)CCC(C)CC1C(=O)NCC(C)(F)C(C)C N1(C(c2c(C)c[nH]n2)=O)CCCC(F)(CNC(c2cc(C)c(O)nn2)=O)C1 C#CC1(C(=O)NCCCC(O)CO)CCN(C(=O)C(C)CSC)C1 C1(CNC(C2C(C)N(C)CC2)=O)CC2(CCN(C(c3csc(Cl)n3)=O)CC2)C1 N1(C(c2c(C(C)C)scn2)=O)CC(C2CN(C(C3(N(C)C)CCSC3)=O)C2)C1 C1(NC(CCc2cn(C)nc2)=O)CCN(C(=O)CN2C(=O)CNC2=O)C12CCC2 C1(C#N)(C(=O)NC2C(NC(C3N(C(C)=O)CCCC3)=O)CC2)CCCOC1 N1(C(C(C)=C(C)C)=O)CCCCC1CC(=O)NCc1nn[nH]n1 c1(C(=O)NC(CNC(c2cc(CC)ncc2)=O)C2CC2)cc(Cl)cc(Cl)n1 Cc1cc(C(=O)NCCCN(C2CCCC2)C(c2cc(C)cs2)=O)c(C)c(C)c1 c1(CC(=O)NC(C)CCCNC(c2c[nH]cc2Br)=O)noc2ccc(F)cc12 c1(C(N(C)CC2CCN(C(C3CC3C3CC3)=O)C2)=O)cc2cccnc2s1 N1(C(C(CCC)C)=O)CC2CC(NC(c3cccn(C)c3=O)=O)CC1C2 C1(CC=C)(C(N2CCOCC2C)=O)CCCN1C(=O)C(O)C=CC C1(C(=O)NC(C=C)C2CC2)C2CCCC2CN1C(c1nccnc1N)=O CC1(C(=O)NCC2(O)CC(NC(c3cc(F)ccc3F)=O)C2)CCC(=O)NC1 C(=O)(C1=CC2CCC(C1)C2)NCc1c(C(N2CC(C)CN(C)CC2)=O)cccn1 c1(OC)cc(CCC(N2C(C(N3CCCC(O)C3)=O)CC3CC23)=O)ccn1 c1(CN(C(C(=O)N(C)CC2CCCO2)=O)CC(F)F)cccc(F)c1 C(C(O)CNC(=O)C(F)F)NC(=O)CCNC(C)=O C1(C2CC2)(C(c2cn(C)nc2)ONC(C2C3CCC(F)C23)=O)CCC1.C1(=O)NO1 c1(C(=O)NC2(CF)CCN(C(=O)CCCC3CCCCC3)C2)n[nH]c2c1COC2 C1(CNC(C2CC(NC)C2)=O)CC12CCN(C(=O)COc1cncc(C)n1)CC2 N1(C(c2c(C)nncc2)=O)CCC2CN(C(c3oc(Br)nc3C)=O)CC12 N1(C(C=CC=CC)=O)C2CCC1(CNC(=O)C(c1c(C)cccc1C)O)CC2 c1(C(=O)NC(CNC(C(CC)C(F)(F)F)=O)(C)C2CC2)ccc2nccnc2n1 N1(CC)CCCC1CC(N1CCC1)=O.C1(NC(C2CCC2)=O)CCCC1F c1(OCC(CC)NC(=O)CCCNC(c2[nH]ccc2CN)=O)ccccc1C C1(COC)CC(O)CN1C(C1CCOC1CNC(c1ccsc1Cl)=O)=O C(C)(CCCC(=O)N1CCC(C)(CN(C)C)C1)NC(c1ccc(C(C)=O)o1)=O Cc1cc(CCC(N2CCCC(CNC(=O)C(C)(C)c3cncs3)C2)=O)n(C)n1 c1(C(N(C2CCN(C(=O)CCCSC)C2)CCC)=O)occ2c1CCCC2 C1(NC(C2C3CCCC23)=O)CC12CCN(C(=O)CCn1cnc([N+](=O)[O-])c1)CC2 Cc1csc(C(=O)NCCC(O)CNC(=O)CCc2ccccn2)c1 C1(CNC(C(C)P(C)(C)=O)=O)CN(C(=O)C=CCN2CCCC2)CC12CCC2 C(=O)(C1=NOC(C)C1C)NCC1CN(C(c2c(C)n(C)c(C(C)C)c2)=O)C1 CC1(C)CCN(C(=O)CP(C)(C)=O)CC1C(=O)NCC=C(Cl)Cl N1(C(CC(=O)NC2CC2)=O)Cc2[nH]nc(C(=O)NCCF)c2C1 N1(CC2CC(O)(CO)C2)CCOCC1CC(=O)NC(c1c(CC)ocn1)=O CC1CC(NC(C2CCC(F)CC2)=O)CN1C(c1cccc(-c2nnco2)c1)=O C(=O)(C(CC1CCCC1)NC(=O)C(F)C1CCCC1)NCC(C)N(C)C c1(CN(C(=O)C=Cc2ccccc2)C)ccccc1CNC(=O)CC1CC1(Cl)Cl C1(CCNC(C(C)NC(N)=O)=O)CN(c2ncc(I)cn2)CCS1(=O)=O C(CCCCCC(=O)NCC1CCCC2CC12)NC(c1n(C)c(O)nc1)=O N1(C(C(COC)(C)OC)=O)CC2(CNC(=O)C(C)(Cl)Cl)CCC1CC2 C1(C(N(C2CCCC2C#N)C)=O)CN(C(C2CC(CF)C2)=O)CCO1 c1(N2CCC(N(C)C(C3CCCN3C3CC3)=O)C2)ncnc2c(Br)nn(C)c12 C=CCC(C)(C)CC(=O)N1CCCC(C)(C)C1CNC(c1cc(=O)n(C)o1)=O C(CC(C)C)(C(=O)NCC(C)C)NC(COC)=O N1(C(C2N(CC)CCCC2)=O)C(CC(=O)NCC2OCCC2C)C2CCCC12 N1(C(CC(CCCC)O)=O)CCC2(CCCN2C(=O)C(C)c2ccsn2)CC1 n1(CC)ccc(C(=O)NCC(C)(CO)NC(=O)CN(C)C)c1C C1(NC(c2cc(C(F)F)ccc2O)=O)CC2(CCN(C(C34CCC3C4)=O)CC2)C1 CC1ON=C(C(=O)N2CCN(C(=O)CNC(C3CCCCC3)=O)CCC2C)C1C Cn1ncc(Cl)c1C(=O)NC1CCC(CNC(=O)C(O)CN(C)C)CC1 C1(C(=O)NCC(C#C)OC)CCN(C(=O)C=C(C)C(C)C)CC1(C)C Cc1ncc(Cl)c(C(=O)NC2CCC(NC(C3CC34CC4)=O)C2)n1 N1(CC(=O)N(CCOC)N)CCCC(NC(=O)OC(C)(C)C)C1.C#CCOC C#Cc1ccc(C)c(NC(C2C(C)CCN2C(=O)CCc2cccn2C)=O)c1 CC(CCNC(=O)CCc1cccc(F)c1)CCNC(C1CC1(C)C(F)F)=O c1(OC)ccc(I)cc1C(=O)NC1CN(C(c2cncnc2)=O)CC1(C)C CC(C1CCCCC1)=CC(=O)NC(C)(C)C(C)NC(=O)C(O)Cn1cncn1 N1(C(c2ccn(COC)n2)=O)CC2CCC(C1)N2C(c1cncc(C2CC2)c1)=O CCC(CC)CC(=O)N(C1CCC(NC(c2cccc(C(=O)OC)c2)=O)CC1)C Cc1ccc(O)c(C(C2CC2)NCC2(C(=O)N(CCO)C3CC3)CCOC2)c1 CON=CC(=O)N1CCC(NC(=O)C(C)(C)C2CCCO2)C1 c1(C(N(C)CC2CCN(C(CCC(=O)NCCC)=O)CC2)=O)cc(C)cc(Cl)c1 N1(C(COCc2c(C)cccc2)=O)CCC(NC(=O)CN=S(C)(C)=O)C(C)C1 Cc1cc(C)c(C(N2CC3C(C2)N3C(=O)C(C)C(O)C(C)C)=O)cc1N C12(C(=O)NC(CNC(C(C)(C3CC3)OC)=O)C)CCCC1C2(F)F C1(NC(c2cnccn2)=O)CC2CCC1CN(C(C1CSCCS1)=O)C2 c1(OC)cc(C(c2nnnn2C(C)(C)C)NCc2nc(C3CCC3)no2)nn1C C(CCC[Si](C)(C)C)NC(C=CCCc1ccn(C)c1)=O C1(C(=O)NCC2C(CNC(=O)CCC3OCCO3)C2)CC2C=CC1C21CC1 C1(NC(C(c2cccc(O)c2F)(C)C)=O)CN(C(C2CC2F)=O)CC2(CCC2)C1 N1(C(C2CC(OC)(OC)C2)=O)CCC(CC(=O)N(CC(F)(F)Cl)C)CC1 N1(CC(=O)NC2CC2NC(c2nc(Cl)sc2Cl)=O)CCCCCC1=O c1(C(=O)N)cnc2c(Cl)cccn12.N1(C)C(C)CCCC1C.CC1C(C)(C)N1 Cn1nc2c(c1C(=O)NCC1COCCN1C(=O)CC1CCC(=O)N1)CSCC2 c1(NCC(=C)Cl)cc(Br)ccc1S(=O)(=O)NC1CCOC(c2ccncc2)C1 c1(C(=O)NC2C3CCN(C(C(F)=C(C)C)=O)C3C2)cnc2c(c1)COC2 c1(C(=O)NC2CCC(C)(CNC(C3(CCOC)CC3)=O)C2)cccc2[nH]ncc12 C(=O)(CCCCN=[N+]=[N-])N1CC2C(CC(=O)NC(c3nc[nH]n3)CC)(CC2)C1 c1(OC)ccc2[nH]c(C)c(C(=O)N(C)CCN(C)C(C3CCCSC3C)=O)c2c1 C(F)(C(=O)N(CC(CCC)NC(CSCC(F)C1CCC1)=O)CC)=CCC Cc1cccc(C(N2CCCC(NC(=O)CC3CCCCC34CC4)CC2)=O)c1O N1(C(C2(CCC)CCN(C(=O)OC(C)(C)C)C2)C(=O)O)CC(C)CS1(=O)=O C1(CNC(C(c2c(C)cccc2)C)=O)CN(C(c2nocc2C)=O)CC1(C)C C1(C(=O)NC(C2CN(C(=O)CC(C)(C)O)C2)C)CCC2(CC1)CC2 c1(C(=O)NCCCCNC(c2c(OC)cncc2)=O)cn(C)c2c(Cl)cccc12 N1(C(CCC=C)=O)CCC(C)C1CNC(c1cnccc1OC(F)(F)F)=O N12CC3CC1CC3C1C(C2C(=O)NCCCSCC)C1.c1(CC)cc(C)nn1C C1(C(=O)NCC(CNC(=O)CC2CCCCC2)OC)CCCN(C(C)=O)C1 c1(SCC(=O)NC2CC(NC(=O)CCC=CBr)C2)ccccc1[N+](=O)[O-] C1(C(C)(C)C)CC(NC(C(=O)NC(=O)C(C)=C(C)C)=O)CCO1 c1(C(N2CCC(N(C(C3CC(OC)C3)=O)C)C2)=O)cccc2c1COCC2 c1(C(=O)NCCNC(CSCC(=O)OCC)=O)csc(CC)n1 c1(OC)ccc(C(=O)NCC2(C)CCCN(C(=O)CC=C(C)C)C2)nc1N N1(C(C(C)=C(C)C)=O)CCC(CNC(=O)Cc2sc(O)nc2O)C12CCC2 C(CC(F)CN=[N+]=[N-])NC(=O)NC(C=CC(=O)N(C(C)(C)C)C)(C)C C1(NC(C2N(C(=O)OC(C)(C)C)CC(C)OC2)=O)CCOCC12CCC2 C1(C)(CNC(CCCC=C)=O)CN(C(=O)C(C)(C)N2CCCCC2)CCO1 C(=O)(CC(C)Oc1ncc(C(N2C(NC(C3CC3)=O)C2)=O)s1)N(CCOC)C C1(C(N2CCC(N(C(=O)CC3CC(C)(C)C3)CC)C2)=O)CC(=O)OC1(C)C N(C1CS(=O)(=O)c2ccccc21)C(c1nc(-c2ccc(CC)s2)sc1)=O C1(c2nn[nH]n2)N(Cc2onc(-c3ccc(C)cc3)n2)CCC1(C)C C=CC1COCCN1C(=O)CCN(C)C(C1CCC(=O)C1)=O C=CC(C)(C)CC(=O)N1CCCC1C(C)(C)CNC(=O)CCCC1CC1 C=C(C)CC(=O)N(CC(CC)NC(C1CCCC1)=O)C N1(C(C)C(=O)N(C)C)CCCC(NC(c2ccc(C(=O)NC3CC3)[nH]2)=O)C1 N1(C(CC(C)(C)OC)=O)CC(C)N(C(=O)Cn2ccc(C(=O)OC)n2)CC1C Nc1c(C(=O)NCC2C3CN(C(c4ccccc4C(F)F)=O)CC23)ccnc1Cl C1(N(C(c2ccc(C)n2C)=O)C)CN(C(=O)C(O)C2CCCC2)CC1(C)C CC(C(=O)NN1CCCC1C(=O)N=c1ccn(C)[nH]1)C1CC1.CNC c1(Nc2ccc(C(CF)OC)cc2)ccc(C)cc1.C12C=CC(C1)NC(=O)NC2 C1(C2CCN(C(C3COC(=O)N3)=O)C2)(NC(c2ccc(OCC=C)cc2)=O)CC1 C1(CN(C(c2n(CC)c(O)nc2)=O)C)CCCN(C(C2(Cl)CC2(C)C)=O)C1 C1(C(=O)NC(CC)(C)CNC(=O)Cn2ncnn2)CNC(=O)C(C)(C)C1 n1(CC)nnc(C)c1C(=O)NC1COCC1CNC(C1C(C)(C)C1(F)F)=O C(=O)(C1CCc2cccnc21)N1CC(O)(CN(C(=O)CCC2CCOC2)C)C1 CS(=O)c1cc(C(=O)NC2CC(O)(CNC(C3CCC3)=O)C2)ccc1Cl C1(C(=O)NC(C2(O)CN(C(C3CC4CCCC34)=O)C2)C)(COC)CCOCC1 Cc1cc(C(N2CCC(C)(NC(c3nnsc3C)=O)C2)=O)ncc1C#N N1(C(C2CN(C(C)=O)C2)=O)CCC(NC(C2(C)CC3CCC2C3)=O)C(F)C1 CC(C)(CCS(C)(=O)=O)NC1CC2CC1CC2O CC(C(=O)NCCCCC(C)NC(C1CCC2(CCC2)O1)=O)S(C)(=O)=O CN1CCN(C(=O)C2=COCCO2)C(CNC(=O)C=Cc2ccncn2)C1 N1(C(C2(C#C)CN(C(=O)CN=[N+]=[N-])C2)=O)CC(=O)N2CCCC2C1 C(=O)(C(C)C(O)C(C)CC)N1CCOCC(F)(CNC(CC2(C=C)CC2)=O)C1 C(=O)(C1CCCc2nc[nH]c21)NCC#CCNC(C1=NOC(C)C1)=O C1(NC(=O)CCC(F)F)CCOC2(CCN(C(c3cn(C4CC4)nn3)=O)CC2)C1 C(C(C)(O)C(=O)N1CC(C(C)NC(c2ccccc2SC2CCCC2)=O)C1)OC c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)C3C(C2)C3)ccc2c(c1)CCC2 N1(C(C=CC2N(C(c3n[nH]c(CC)c3C)=O)CCC2)=O)CCCC12CCCC2 N1(C(CCC=CCC=C)=O)CC2CC2(NC(=O)CSc2ccccc2Cl)C1 C=CCCC(C(=O)NC(CO)C(C)C)NC(=O)CN(C)CC N1(C(c2csc(C)c2C)=O)CC(C)(C)CC1CNC(c1ccc(C(N)=O)s1)=O CC1(C)C2CC(CN3CCCC3(C)C3CCC3)CC12 C1(C(=O)NCC2CC(NC(C3CCCC(F)C3)=O)C2)(CC)CCC(O)CC1 c1(C(=O)NC(CNC(C2(C=C)CC2)=O)C)coc2c1NC(=O)CCC2 N1(NCCC(CC)(O)CC)CCC2(CCCCC2CN)CC1.C(=O)N(C)C ClC(Cl)CN=c1[nH]c2c(c(=NCCN3CCOCC3)[nH]1)CSC2 C1(NC(c2cn(C(C)C)nc2)=O)CCC12CCN(C(=O)CN1CC3CC3C1)CC2 c1(C(N2CCN(Cc3cccc(OC)c3)CC2)C(=O)NCC)cccnc1C C1(CNC(CSC(C)C(N2CCCC2)=O)=O)N(CC2CCCO2)CCC1(C)C c1(C(=O)NCC(CNC(=O)C(F)=C(C)C)OC)c(Cl)sc(C)c1C C(C(=O)NC(C)C(=O)NCC(F)C(C)(C)O)(C(C)C)SC Cc1noc(C)c1C(C)C(N1CCC(Cn2cc(CC3CCOC3)nn2)CC1)=O O=C1OCC2CCN(C(C3CC(NC(=O)Cc4ccsn4)C3)=O)C12 c1(C(=O)NC2CN(CC(CCC)O)CC2n2ccnn2)cn2cc(F)ccc2n1 c1(NC(C(CCCOC)NC(C2OCCC2(C)C)=O)=O)cnc2ccnn2c1 C12(NC(C3N(C)C(=O)CC3)=O)CCOCC1CN(C(c1cc3scnc3[nH]1)=O)C2 CCCCC(=O)C(=O)N1CCC(CCNC(c2c(F)cccc2F)=O)C1 CC1CN(C(c2ccoc2)=O)CCC1CNC(=O)CC1(N(C)C)COC1 C(=O)(C(C)(C)N=[N+]=[N-])NCC(CC(=O)N(CC(C)(C)O)C)O c1(CC)cnc(C(=O)N(CC(=O)NC2CC3(CSC3)C2)CC2CC2)nc1 c1(OC)cc(C(=O)NC2CC(C)N(C(=O)CSC(F)F)C2)cc(N)c1N C1(C(=O)NCC(COC(C)C)O)CN(C)CCN1C(c1cnc(O)n1C(C)C)=O C1(C(=O)NC2(CC)CN(C(c3cnn(C)c3)=O)C2)CCCC(C(=O)OC)CC1 C1(C(N(CCCC)CC(=O)NCC(C2CCCCC2)C)=O)Cc2nccn2C1 N1(C(C(CCCC)O)=O)CC2CCC1C1CN(C(c3cccc(Cl)c3O)=O)CC21 c1(C(=O)OC)ccc(NCC2CCC(C(=O)NCCC3CCN(C)C3)C2)nc1 C(C(C(C)(C)C)NC(=O)C(C)(C)N(C)C)NC(c1ccc(CC)o1)=O N1(C(C=Cc2n(C)ncc2)=O)CCC2CN(C(c3nocc3Cl)=O)CCC2C1 c1(C(N2CC(C)C(NC(c3cccc4nonc34)=O)C2)=O)cc2ccncc2s1 c1(N(CC(=O)NCC#C)C)cc2cccc(N)c2cn1 N1(C(c2[nH]cc(C)c(=O)c2)=O)CCN(C(C2CCCCC2F)=O)CC(C)C1 c12cccc(c1)O2.C1(C(=O)OCC)CCCN(C(C)=O)C1 N1(C(COC(CC)=O)=O)CC2(C)CC1(C(N1CC3CC3C1C(=O)OC)=O)C2 C=C(Cl)CCC(=O)NC1C(C(N2CCCC2C(C)(C)CO)=O)C1(C)C N1(C(Cc2nc(CC)sc2)=O)CCOCC1CN(C)C(C1(C)CCCOC1)=O N1(C(C2N=C(C)SC2)=O)CCC(NC(=O)C2=CCCCC2C)C(CO)CC1 C(=O)(C1=C(C)CCCC1)NCC(CN(C(c1cnc(OC)nc1)=O)CC)(C)C N1(C(CC(C=C)c2ccccc2)=O)CCN(C(C2CC(C)C2)=O)C(C)C1 N1(C(c2c(COC)noc2)=O)CCC(C)C1CNC(C1(OC)CCC1)=O C(CC(C(=O)N1CCN(C(C2CC=CCO2)=O)CC1)NC=O)SC C1(C(=O)NC2CN(C(C(C)(Cl)Cl)=O)CC2F)CC(S(C)(=O)=O)C1 N1(CCOC)C(C)CN(C(c2cccc(C#N)c2)C(=O)NC2COC2)CC1C c1(C(N(C(CCNC(C=C(COC)C)=O)C)C)=O)ccc(C2(F)CC2(F)F)cc1 C1(CNC(c2cc(COC)oc2C)=O)COCCN(C(=O)CCC=C(C)C)C1 c1(CC)noc2ncc(C(=O)NC3CC4CN(C(=O)Cc5cc[nH]c5)CC34)cc12 Cc1ccccc1C1(NC(C2CC(c3cccc(Cl)c3)(O)C2)=O)CCC1 C1(NC(c2cc(COC)on2)=O)CN(C(=O)CCc2nc(C)no2)CC(C)(C)C1 C(=O)(CC(O)CC(C)(C)C)N(C1CCCN(C(C2CC(SC)C2)=O)C1)C c12ccc(cc1)Cn1nnnc1C2OCC.C(CC(C)(C)C)NCCOC(C)C CC(CF)N=c1ccn2ncc(S(=O)(=O)N3CCOC(CS(N)(=O)=O)C3)c2[nH]1 CS(=O)(=O)c1ccccc1CC(N1CCC(CCNC(=O)CCCCCF)C1)=O N1(C(=O)C=Cc2cccs2)CCC(CNC(c2c(O)cccc2F)=O)C(F)(F)C1 C1(O)(CCNC(C2(CCOC)CCC2)=O)CN(C(=O)C(C)C2CCC2)C1 N1(C(C2C(C3C(C)C3)C2)=O)CCN(C(=O)CCF)CC(C)(C)C1 c1(NC(c2ccc3c(c2)CN(C)C3)=O)ccc2c(c1O)CCCC2 c1(C(=O)NC2C(C)N(C(c3ccc(C(C)(C)C)nc3)=O)CC2)ccc(F)cc1F C1(NC(CC=C)=O)CN(C(=O)CC=Cc2ccccc2F)CCC1CO c1(C(=O)NC(CCN(C(CC(C=C)CC)=O)C)C)ccn2cc(C)nc2c1 Cn1ncc(C(N2CC(n3cc(C4(C(N)=O)CC4)nn3)C(O)C2)=O)c1C#N Cc1cccc(Cl)c1C(N1CC(NC(c2cncc(Cl)c2)=O)C(C)(C)C1)=O c1(C(=O)NC2CN(C3COC3)C2)ccc(Br)c2c1OCCC2 c1(C(=O)NCCOCCNC(c2cc(C)on2)=O)nc(Cl)c(Cl)s1 C1(NC(CN(CCOC)C(C2CC(=C)C2)=O)=O)CCCC(O)C1O C(CC(O)C(=O)NC(C1CCOC1)C)NC(Cc1cnc(C)s1)=O C(N=C(NCc1ccccc1)N(C)CC1(N(C)C)CC1)c1c(C)nc(C)s1 c1(C(N2CCC(C(N3CCC(COC)C3)=O)(CF)C2)=O)cccn(C)c1=O c1(CC(C(=O)NCC(CC)NC(=O)C(C)CC(C)C)C)ccc(F)c(Br)c1 C1(C(N2CC(CC=C)(NC(c3ccc(Cl)cc3CC)=O)C2)=O)CCCC(C)CC1 N1(CCCOC)CCC(N=c2[nH]c(N(C)Cc3c[nH]c(Br)c3)nc3c2COC3)C1 C(=O)(C#CC1CCOC1)N1CCC(C(CNC(Cn2c(C)nnn2)=O)(C)O)CC1 C(CC(=O)NC1CSC1)OCCNC(CSC(C)C)=O C1(F)(C(=O)OCC(=O)Nc2n(C)cnn2)CC=CCC1 N1(C(c2c(C)nc(C)s2)=O)CC(C)CN(C(C2CC3C=CC2C3)=O)C(C)C1 CC1=C(COC(=O)C2=NNC(C(F)(F)F)C2)C(C)(C)CCC1 c1(C(N2CCCN(C(CC3C(C)CCCC3)=O)CC2)=O)ccc(Cl)cc1F c1(C(=O)NC(C)CCNC(=O)CNC(c2cccs2)=O)cccc2c1CCN2 N1(C(C(C(CC)C)N)=O)CCC2CN(C(=O)C(c3ccc(C)cc3)C)CC2C1 CC1(C)CCN(C(C2CCOC2(C)C)=O)C1C(=O)NCc1ncc[nH]c1=O CCCN=C(NCc1cc(C)on1)NCc1cc(C2CC2)on1 CC(C)CC(C(=O)NCC1CCC1CO)ONC(C1(C)CCC(=O)C1)=O c1(C(N2CC3C(C(=O)NC(c4cn[nH]c4)C)(C3)C2)=O)ccc2nc(Cl)ccc2c1 N1(C(c2cnc(OC)nc2)=O)CC2CC(C(N3CCOCC3C(C)O)=O)(C2)C1 N1(C(=O)C(c2ccccc2)F)CC2(CC(C(=O)NCC(=O)NC3CCSC3)C2)C1 C1(C(N2CCC2C2CCCCC2)=O)(CNC(=O)CCN2CCCC2)CCOCC1 C(=O)(C(O)CC(F)(F)F)NCC1(OC)CCN(C(c2cc3ccncc3s2)=O)C1 C=C1CN2C(=O)CCC2(C(N2CCC2CNC(=O)COc2cccnc2Cl)=O)C1 C(=O)(C(CC(F)F)NC(c1coc(OC)n1)=O)N(CC(CC)OC)C Cc1csc(C(N2CCCC(C(=O)Nc3cn(C)nc3C)C2)=O)c1C c1(NC(C2N(Cc3ccc(C)cc3C)C3C(C2)C3)=O)cc(C)c(Br)c(C)c1 N1(C(C(C)OC2CCOC2)=O)CCCC(NC(C2(C)COC2)=O)C1C N1(C(C2(C)ON=C(C)C2)=O)CCCC2(C1)CN(C(C1OC(C)CC1C)=O)CCO2 N1(C(C2=C(CC)OCCS2)=O)CCC(C2CCN(C(=O)CN3CCOCC3)C2)C1 N1(C(CCc2ncc(C)[nH]2)=O)CCC2(CC1)CCN(C(=O)C(C)CS(C)=O)C2 C1(C(N(CC(C)C)CC#C)=O)CN(C(=O)C(c2ccn(C)c2)C)CC1(C)C c1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)no2)=O)cn2c(n1)SCC2 c1(C(N2CC(C)(NC(=O)CC3(C)CCS(=O)(=O)N3)C2)=O)cc(Cl)c(F)cc1O C1(C(N(C)CC2CC2(C)C)=O)N(C(c2cnn[nH]2)=O)CCC1(C)C CC1CCn2cc(C(N3CCCC(NC(c4cccc(Cl)n4)=O)C3C)=O)nc2C1 C#CCC(C(=O)NCC(C)(C)CC1CC1)NC(=O)C(C(C)C)C1CCC1 C1(CC(N2C3CN(C(c4n(C)ncc4)=O)C(C3)C2)=O)Cc2cccc(Cl)c2O1 C(C(=O)NCCCC1CCCN1C(=O)CCn1ccnc1)(C(C)C)OCC(C)C N1(C(CCC(=C)Cl)=O)CCC2CCN(C(c3nn[nH]c3Cl)=O)CC12 c1(-n2ccc(C)n2)n[nH]c(=NC2CC(NC(=O)C(F)C(C)C)C2(C)C)s1 Cc1c(F)ccc(C(N2CC3CN(C(=O)C(F)=C4CCC4)CCC23)=O)c1C c1(NCC(CCCC)NC(C2CCN(C)C2=O)=O)nc(Cl)nc2[nH]cnc12 c1(-c2onc(-c3c(-c4n(-c5ccc(Br)cc5)nnc4)csc3)n2)cn2c(n1)CCC2 Cc1ccnc2nc(C(=O)NCCCCCCNC(C3CCNC3=O)=O)nn12 Cc1ccc(C(N2CCN(C(=O)C(O)C(C)C)CC2C(C)C)=O)cc1CC(C)C Cc1cc(C(=O)NC(C)CCCNC(=O)C(C)NC(=O)C2CC2)cc(N)c1Cl N1(S(CCOCC)(=O)=O)CCCCC(C(C)OC)CC1 C1(C(=O)NC2C(NC(c3cc(Br)c[nH]3)=O)CC2)Cc2cncn2C(=O)N1 CCC(CC)CC(F)C(=O)N1CC(NC(c2cncnc2)=O)CC(F)C1 c1(NCC(=O)N(C(c2cccc(OC)c2)C)C(C)C)c(Cl)cc([N+](=O)[O-])cc1Br C1(NC(CCOC)=O)CCN(C(c2cc(N)cc(O)c2)=O)C(C)C1 C(=O)(C(C)CC1CCCCC1)N(CCC(C)NC(c1coc(C2CCC2)n1)=O)C C1(C(=O)NC2CCCN(C(c3csc(C)c3C)=O)C2)SC2C=CC1CC2 C1(NC(CCN(C(CC2N(C)CCCC2)=O)C)=O)CCCN(C)C1=O Cc1cc(F)ccc1N(C(=O)C(CC(C)C)ONC(c1ccc(F)s1)=O)C CCC(C(=O)OC)C(=O)N1CSCC1C(=O)NC1(C)CCC(C)(C)C1 C12(CNC(c3c(C)noc3N)=O)CCCCC1N(C(=O)CN(C)CCO)CC2 c1(C(N2CC3C(NC(C(N4CCC(C)C4)=O)=O)(C3)C2)=O)ccnc2ccnn12 C1(CC=C)(C(=O)OCC)CCCN(C(CC2CCOCC2)C(=O)NC(C)CC)C1 C(CCCC(CO)NC(=O)C(CO)C(C)C)NC(CN(CCC#C)C)=O c1(OC)ccc(S(=O)(=O)N2CC=CC2C(=O)Nc2ccc3nc(C)[nH]c3c2)cc1F c1(C(N2CCC(C)C(NC(=O)CSC(F)F)C2)=O)cc2cccnn2c1 CCC(C(=O)N1CCN(C)C(CNC(C2CNC(=O)O2)=O)C1)C(C)(C)CC c1(C(=O)NC(C2CCN(C(CCOC)=O)CC2)(C)C)ccc2nc(OC)[nH]c2c1 c1(C(N2CCCN(C(CC(COC)C)=O)CC2CO)=O)c(Cl)nc2ccccn12 n1(CCCOC(=O)COc2ccc(Br)cc2)cccnc1=O N1(C(CCCOC)=O)CCN(C(c2ncc(C(F)F)s2)=O)C(C(C)(C)C)C1 c1(OC)cc(CCOC(c2ccnc(SC)n2)=O)ccc1OC N1(C(CCCNC(=O)OCC)=O)CC(NC(=O)C=CC=C(Cl)Cl)CC(C)(C)C1 CCCCCC(C)(C)C(=O)NC1CC(NC(=O)Cc2cc(F)ccc2Cl)C1 C1(NC(C2CC3(CC(=O)N3)C2)=O)CCCC12CCN(C(C1CCS1(=O)=O)=O)CC2 c1(CC(=O)N(c2ccc(OCC(F)F)cc2)C2CC2)cc(F)cc(Cl)c1 C(=O)(CC(C)C(C)(C)NC(=O)C(F)n1ccnc1)NCc1ccc(C)nn1 N1(C(N2CC(C)C(OCc3ccccc3)C2)=O)Cc2c(Cl)cccc2C(C)C1 C12(NC(C3CN(C)C3)=O)CCC1CN(C(c1ccc(OCC(N)=O)cc1)=O)C2 C(=O)(C(CNC(=O)C(C1CC1)SC)CC1CC1)NC(CCOC)CO C1(C(=O)NC2C(SC)COC2)CCCCCCN1C(=O)CCCC1CCCC1 C1(C(=O)NC2CCC(CC)CC2)CN(C(n2cnnn2)=O)C2(CCC2)C1 c1(C(=O)N(C(C)CCNC(c2cccc[n+]2[O-])=O)CCO)cc(O)nc(C2CC2)n1 CCC(O)(C(=O)NCC(=C1CN(C(=O)CC2(C)CC2(F)Cl)C1)F)c1ccccc1 CCCCC(C(=O)NCCOC1CN(C(C2CCOC2=O)=O)C1)C(C)C C1(N(C(c2occ(C)c2)=O)C)CCC(NC(C2CC2c2ccsc2)=O)CC1 C(=O)(CC(C)(C)C)NCC1OCC(C(=O)NCc2ncc(CC)s2)C1 c1(CC)ccc(C(N2CCN(C(C3CN(C)C3)=O)C(CC)C2)=O)c(Cl)c1 C(=O)(C(O)CCC(C)C)N1C(CNC(C(CC)N(CC)CC)=O)CC(OC)C1 c1(OC)cnc(N(Cc2cnn(C3CNC3)c2)CC2CN(C)CCO2)nc1C C1(C)(COC)CC(NC(=O)CCSC2CCC2)CN1C(c1c[nH]cc(Cl)c1=O)=O C1(C(N2CC(n3ccnc3)C2)=O)(N(C2CCOC2)C(C2CCSC2)=O)CCC1 Cc1c(Br)ccc(-c2noc(C(=O)Nc3cccc(F)c3Br)n2)c1F O=S(=O)(c1ccc2[nH]c(=NC3C=CCCC3)sc2c1)NCCn1nccn1 O=C(C(O)CC(F)F)NCC1(F)CCCN(C(C2(C(N)=O)CC2)=O)C1 Cc1ccc(CN2CCN(C(=O)N(c3[nH]cnc3CO)CCO)C(=O)C2)c(C)c1 C12(NC(c3n(C)c(S)nc3)=O)CCC(CC1)N(C(C1CCC3C(C1)C3(F)F)=O)C2 N1(Cc2c(C(=O)O)c3c(s2)cccc3)CC2CS(=O)(=O)CC(C1)C2(F)F c1(C(=O)NCC(C)(C)CNC(=O)CCn2cc(Cl)cn2)c[nH]c(=N)nc1O C#CC1(C(=O)NCC2CC(C(C)C)C2)CCN(C(=O)C=C(C)C(C)C)C1 c1(-c2cn(C3CCN(C(C4CCS(=O)(=O)C4)=O)C3)nn2)ccc(F)nc1 C1(NC(c2n[nH]cc2F)=O)CN(C(c2cnn3c2CCC3)=O)CC12CCOCC2 N1(C(c2c(OC)c(C)ccc2)=O)C2CCC1CN(C(=O)CN(S(C)(=O)=O)C)CC2 c1(CC#C)nc(C(=O)N)co1.C12(OCC)CN(C1)C2=O.c1(OC2CC2)ccccc1 CC1(CNC(C2CCC(OC(F)F)CC2)=O)CCCN(C(=O)CSC2CC2)C1 c1(C(N2C(CCNC(C(CC)N(C)C)=O)CCC2)=O)c(OC)cc(OC)cc1F Cc1ncc(C(=O)NC(C2CN(C(c3cc(C(C)C)on3)=O)C2)C)n1C N=C1NC(=O)C(CC(N2CCN(C3CCCN(C(=O)CC4CC4)C3)CC2)=O)S1 CC1CN(C(c2cscc2C#N)=O)CCC1CNC(C1CCCC12CC2)=O S(=O)(=O)(c1ccc(Cl)c2nonc12)NC(C1C(NC(=O)Cc2ccc(Cl)cn2)C1)=O C1(NC(CS(CCOC)(=O)=O)=O)CCC2CN(C(C3CCC(=O)N3)=O)CCC2C1 c1(C(=O)NCC2C(NC(c3ccsc3CO)=O)CC2)ccc2c(c1)CCNC2=O N1(C(CCNC(Cc2cn(C)nc2)=O)=O)CC2CCC2C1 N1(C(C=C)=O)CCC2(CCCC2NC(c2cc3c(C)cccc3o2)=O)CC1 c1(OC)cc(N2CCC(C)C(NC(C3CC(C)CO3)=O)C2C)c(Cl)cc1[N+](=O)[O-] CC(C)C(C(=O)NC1CCCC1CC(=O)N(CC(C)C#N)C1CC1)C1CCC1 C1(CNC(=O)CCc2ncccn2)CCC2(CCC2)CN1C(=O)C=CCF C(=O)(CC(C(F)F)SC)N(C(CNC(Cc1ccc(C(=O)OCC)cc1)=O)C)C Cn1ccc(=O)c(C(=O)NC2CC(C(=O)NC3CC34CCC4)C2)c1 C1(C(N2CCC(C)C(NC(c3ccc(=O)n(C)c3)=O)C2)=O)CCCC2(CCC2)C1 C1(CNC(C(C)C2CCOC2)=O)(NC(C2(F)CCCCC2)=O)CCC(C)(C)CC1 N1(CC(N2CCCCC2c2nc[nH]n2)=O)CCN(Cc2ccc(F)cc2)CC1=O N1(C(C2CC(F)C2)=O)CC2=C(C1)CN(C(C13CCCC1C3)=O)C2 C1(C(=O)NC(CC)CC)C(C)CCN1C(=O)C(C)NC(=O)C1CC1 c1(C(=O)NCC2CC(CNC(c3cccc(C)n3)=O)C2)cnc(C)c(N)c1 c1(CC)cc(Cl)ccc1N.N1(C(=O)C(=O)NC2CSCC2OC)CCCC1CO C1(C)(OC)CC2CC1CC2NS(=O)(=O)CC1CC2(C1)CC2F N1(C(c2nccn2C(F)F)C(=O)NC2CCCC2)CCCNC(CC(F)(F)F)C1 C1(CC)CCN(C(C2(NC(c3cccc(C)n3)=O)CCCC2C)=O)CCO1 Cc1csc2nc(CC(=O)NCC3(O)CC(CNC(C45CC(F)(C4)C5)=O)C3)cn12 c1(NC2C(C)CS(=O)(=O)C2)nc2c(c(=NCC3Cc4ccccc4C3)[nH]1)CCC2 C1(CNC(CNC(N)=O)=O)CN(C(=O)COc2cncc(Cl)n2)C2CCCC2O1 N1(c2nc(C)cc(OC)n2)CC(NC(=O)CC(C)(O)C2CC2)CC2(CCC2)C1 c1(S)ccc(C)cc1.n1(CCSC)nnnc1C1(NCC2CSC2)CCC1CC(C)C Cc1cc(C)c(CN2CCC(n3cc(CNC(C4CCCO4)=O)nn3)C2)s1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC)CCCNC(=O)CCCN1CCCC1 N1(C(c2cc(=N)[nH][nH]2)=O)CCOCC1C1CCN(C(=O)Cc2ncc(Cl)s2)C1 C1(CNC(=O)COC2CCCCC2)C(C2CC2)CCN1C(=O)C(F)C1CCC1 c1(C)cn(C)c(=O)nc1O.CC1CC(C)N(Cc2c(O)cccc2)C1 c1(C(N(C2CCCC2)CCCNC(C2(C)ON=C(C)C2)=O)=O)cccc(N)c1O C1(NC(C2CC(C#C)(O)C2)=O)(CNC(C2CC3CCC2O3)=O)CCCCCC1 CC(C)CCC(O)C(=O)N1CCC2(CC2)CC1C(=O)NCC=C(Cl)Cl c1(C(=O)OC)cc(N2CCC(CNC(C3CCOC3)=O)C2(C)C)nc(Cl)n1 c1(CN(C(c2cnn(C(F)(F)F)c2)=O)C2CC2)cn(CC2(C(F)(F)F)CC2)nn1 c1(C(=O)NCC(C)NC(c2[nH]nc3ncccc23)=O)ccc2c(Br)cnn2c1 Cc1cc(C(N2CC(F)(C(=O)Nc3cccc(N4CCCC4)c3)C2)=O)cnc1O c1(C(=O)NCCOCCN(C(C2C(OC)C2)=O)C)cnn2cc(C)cnc12 C#CCCCC(C)(c1nnnn1C)NC1(C)CN(C(=O)CC)CCO1 Cc1conc1C(=O)NC(CNC(c1cc(-c2ccccc2)[nH]n1)=O)CO c1(CCC)nc(C)c(C(=O)NCC2(NC(=O)C(C)CC3CCC3)CCCC2)s1 Cc1nnccc1C(=O)NC(C(=O)NCC(C1CC1)N(C)C)c1ccoc1 C1(C(N(CC=C)CCO)=O)CCCN(C(=O)CS(=O)CC)C1C c1(C(N2C(CNC(C(CCC)OC)=O)CC(O)C2)=O)sc2ccc(Cl)cc2c1C c1(C(=O)NC2CC3CCC(C2)N3C(C2CCCO2)=O)cc([N+](=O)[O-])ccc1O c1(C(=O)NCC2CN(C(c3cnc(C)s3)=O)C(C)C2)cnc(N)c(CO)c1 N#Cc1cccc(C=CC(=O)NC2(CNC(=O)Cc3ccc(Br)nc3)CC2)c1 C=C(Cl)C(C)(C)C(=O)N1CCC(NC(=O)CSc2c(C)noc2C)C(F)C1 C=CCC(C)(CC)C(=O)NC1COCC1NC(C1(CCO)CC1)=O c1(CNC(=O)NC(C)COC(F)F)ccnc(N2CCCC2)c1 c1(C(N(C)CC2CN(C(C3CC3(C)C)=O)CCO2)=O)cc(C(F)(F)F)cnc1O c1(C(=O)NCc2c(C(N(CC(O)COC)CC)=O)[nH]cc2)ccc(C)nn1 C(CC(=O)N1CCOC2CC12)(C(F)(F)F)NC(C1(C#N)CCC1)=O N(C(=NCC(C)c1ccsc1)NCN1CCOC(C(F)(F)F)C1)CC(C)C c1(C(N(C2CCN(C(c3cc(C)ns3)=O)C2)CCO)=O)cccc(Cl)c1Cl O=C1CCN(C(c2cccc(Br)n2)C(=O)NCc2cccs2)CCN1 CC(c1cccc(C)c1)=CC(N1CCC1CNC(c1cn(C2CC2)nn1)=O)=O N1(CC(c2c(OC)cccc2)OC)CC(=O)N(CC2(C3CCCCO3)CC2)C1=O c1(OC)cc(C(=O)NCC2CN(C(c3c[nH]c(C#N)c3)=O)C2)cnc1O C=CCCCC(=O)NC(C)CCCNC(=O)Cc1nncn1C c1(CC)cccc(F)c1C(N1CCC(CO)C(CO)C1)=O.C1(=O)C(C)(C)N1 Cc1ccc(N)c(C)c1C(=O)NC(C)CCCCNC(=O)C(C)C(F)(F)F c1(C(=O)NC(C(=O)NCc2c(OC)cccc2)CC2CC2)cc(F)cc(F)c1 c1(OCCC)cc(C(N2CCC(OC(C)C)CC2)=O)cc(OC)c1 N1(C(C(COC(C)C)NC(C)=O)=O)CC2CC(C1)N(C(C1(C)CC=CC1)=O)C2 CC(CCS(C)=O)N=c1[nH]c(=NCCc2ccc(Cl)s2)[nH]c2cccc(F)c12 N1(C(CCC=CCC=C)=O)CC(NC(c2conc2C2CCCO2)=O)C(C)(C)C1 C1(NC(C2CCCC(C)(C)C2)=O)CCN(C(c2csc(Cl)c2Cl)=O)CC12CCC2 CCC(CC)(CO)C(=O)N1CC2CC(O)C1C2NC(c1cc(F)cc(F)c1O)=O N1(C(CNS(NC)(=O)=O)=O)CC23CCCCC2(C1)CN(C(C1(C#N)CC1C)=O)C3 c1(C(N2C(C)CN(c3ccccc3)CC2)=O)c(F)cc(Cl)cc1F c1(C(=O)NC(CN(C(c2cnn(C(C)C)c2Br)=O)CC)C)cnc(NC)cn1 C1(CCOC)(C(N2CC(C)C(F)(F)C2)=O)CCN(C(c2c[nH]nc2OC)=O)CC1 c1(C(N2CCC(CC(=O)NC(C)C(F)(F)F)C2)=O)cc(Cl)nc(Cl)c1F c1(CC)[nH]nc(C(N2CCC(F)(CNC(=O)CCCC3CC3)C2)=O)c1Br C(N=c1nc2sccc2c(N2CCCCC(C)(F)C2)[nH]1)c1nn(C)c(Br)n1 C1(CNC(=O)Cc2cccs2)CN(C(C2(CC(F)(F)F)CC2)=O)CC1C(F)F C(=O)(C(C(C)(C)C)NC(=O)CCCC1CCC1)NCC1(CO)C(C=C)C1 N1(C(CC2(C(=O)OC)CCOCC2)=O)CCCC(CNC(c2ccns2)=O)CC1 C1(NC(=O)NCC(C)CC2CCC2)CCCC1P(C)(C)=O CC1CN(C(C2C3CC4CC(C3)CC2C4)=O)CC2(CCN(C(=O)CC#N)C2)O1 C1(CC)CN(C(=O)C(C)CC(=O)OC)CCN1C(c1cccc(C)c1)=O c1(CCC(=O)NCCC(=C)CNC(c2ccnc(SC)c2)=O)ccc(F)nc1 N1(C(CNC(C(C)(C)C)=O)=O)CCC2(CCC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 C=CCCC(O)CNC(C1CC1C(C)NC(c1c[nH]nc1C(C)C)=O)=O C1(NC(CCN(S(C)(=O)=O)C)=O)COCCN(C(c2cncnc2C2CC2)=O)C1 CC1(C)CCN(C(=O)CCCCN(C)C)C1CC(N1CCCC(O)(C(N)=O)C1)=O CC(C)C(CNC(=O)C=C1CCOCC1)C(=O)NCCCN1CCCC1C c1(NC(C(C)C)C)ccc(S(=O)(=O)NC2CN(C)CC2O)cc1C#N C1(N(C(C(C)OCCC=C)=O)C)CN(C(=O)Cc2c(C)noc2Cl)CC1(C)C C12(C(=O)NC(CC)CC)CC(CN1C(=O)C(C)(C)COC(C)C)C2 CC12CC3CC(CC(C(N4CCCC(O)(CNC(C5CC5(F)F)=O)C4)=O)(C3)C1)C2 c1(C(=O)NC(C)CNC(C2CC3CCC(C2)O3)=O)ccc([N+](=O)[O-])cc1N c1(C(=O)NC(CCCNC(C(C)NC(CC)=O)=O)CO)c(C)cccc1Cl N1(C(C23C(C)(C)C(CC2)CC3)=O)CCCN(C(=O)CN2CC3CC3C2)CC1CO CC(CC(C)NC(=O)C=CCF)NC(c1ccc(C(F)(F)F)o1)=O.N1(C)CCOCC1 c1(CN2CCC(N(C)C)(C(N)=O)CC2)c(C(N)=O)oc2ccccc12 c1(C(C)=O)c(C)[nH]c(C(=O)NCC(C)NC(c2ncc(F)c(OC)n2)=O)c1C C1(CCOC)(C(N2CCC(CNC(c3cnsn3)=O)C2)=O)CCCC1 N1(C(C=COCC)=O)CCC2CC1CN(C(c1sccc1OC)=O)C2 CP(C)(=O)CCC(=O)N1CCC(C(=O)Nc2ccc(C3CC3)nc2)C1 Cn1c(=O)[nH]c(NCCCNC(c2cncn(C)c2=O)=O)c(C#N)c1=O C1(C(N(C(C2C3CC4C(C3)C24)=O)Cc2ccc(CC)cc2)=O)CC(=O)N(OC)C1 c1(NC(=O)CCNCC2NCCC23CC3)ccc2c(c1)CCCO2 C1(NC(C2CCOCC2)=O)CCC(C(=O)NCCc2cn(C(F)F)cn2)CC1 C1(CC)(CC)CC(NC(=O)C(F)C(F)(F)F)CN1C(=O)CC1(COC)CC1 N1(C(C(=O)NCC2C(NC(c3cc(Cl)cs3)=O)COC2)(Cl)Cl)CCCCC1=O C(CC(CC)C(=O)N1CCC(CNC(=O)Cc2ccsc2)C1(C)C)=CC Nc1ccc(CCNC(=O)C(F)CC2CCOCC2)cc1 Cc1noc(N)c1C(=O)NC1CCN(C(c2coc(-c3ccsc3)c2)=O)CC1 C(CC1CCCCC1)(C(=O)OC1CC(CC(N)=O)C1)NC(=O)OC(C)(C)C N1(C(CCC2N(C(c3c(CC)[nH]cc3)=O)CCCC2)=O)CCNC(=O)CC1 Cc1cccc(C(C)C(=O)NCC2CCCN(Cc3ccc(CCN)cc3)C2)c1 N1CC2(CCC(N)CC2)C1.c1(C2(C)CC2)cc(C(=O)NC(=O)CC2CC23CC3)[nH]n1 N1(C(C(C)OC)=O)CCN(C(=O)C(F)(F)CCn2ccnn2)CCC1C Cc1nc(C(=O)NC(C)CCNC(c2coc(Cl)n2)=O)c(C(F)(F)F)[nH]1 c1(NCCC(=C)C)cc(Br)ccc1S(=O)(=O)N(CC(C)C)C c1(C(=O)NCC2(C)CCCN(C(=O)CC3C=CCC3)C2)cc(C#N)ccc1O N1(C(c2c(C)noc2)=O)CCN(C(c2ccc(F)c3ccsc23)=O)CC12CCC2 c1(CNC(C(C)N(C(c2n(CC)ccc2)=O)C)=O)ccc(C)nc1 c1(C(=O)NCC2C(CNC(Cc3cn(C(C)C)nn3)=O)C2)ccc2nn[nH]c2c1 C1(CC(N2C(Cc3cn(CCC(C)C)nn3)CCCC2)=O)SC(=S)N(C)C1=O CC1(CNC(=O)CCOCc2ccccc2)CCN(C(C2CC(O)(C#N)C2)=O)C1 c1(OCC)cc(C)ccc1-c1cn(CCNC(c2ccc(C(C)C)cn2)=O)nn1 C1(CCNC(C(C)Nc2scc(C)n2)=O)CCCN(C(C2(C(F)F)CC2)=O)C1 C1(NC(CCc2c(C)ncs2)=O)CCN(C(C2(COC(C)C)CC2)=O)CC1C c1(CC)ccc(C(=O)NC(C)C(CO)NC(C2(C(F)F)CCC2)=O)c(C)n1 c1(-c2n(CC(=O)OCC)nc(C(C)CCC)n2)cn2cccc(OC)c2n1 C#Cc1ccc(Br)c(C(N2CCC(N(C(=O)CC3CCOC3)C)C2)=O)c1 Cc1nc2c(o1)CCN(C(C1CCCN1C(=O)Cc1noc(C)c1C)=O)C2 C1(NC(C(c2cccs2)NC(CCCCOC)=O)=O)(CO)CC2CCCC12 c1(C(=O)NC2(CCNC(C(C)n3ccnn3)=O)CCC2)ccc(N)c(F)c1F C1(NC(c2c(SCC)cccc2)=O)CCC2(C1)CN(c1ncncc1C(=O)OC)C2 Cc1nn(C)c2sc(C(=O)NCC(C3CC3)NC(=O)CC3CC3C(F)(F)F)cc12 CCC(C)(CNC(c1ncoc1C1CC1)=O)NC(c1cc(C2CCC2)[nH]n1)=O C1(NC(c2cc(-c3cn(C)nc3)no2)=O)CCN(C(C2(C)CC=CC2)=O)CC1O C1(NC(c2c(C)cc(C)s2)=O)CC2CC(C1)N(C(=O)CCCC1CCOCC1)C2 C(=O)(C(C)CC(C)(C)C)NC(CCCC)C(N1CC2(CCC2)CC1C)=O c1(CCCOC)nc(CCc2cnn(C)c2)n(-c2ccnc(Br)c2)n1 C1(O)(CCNC(C(C2CCCC2)OCC)=O)CCN(C(C23CSC(C2)C3)=O)C1 C1(C)(CNC(C(C)Cc2cccnc2)=O)CCN(C(C2CCCC2)=O)C1 S(=O)(=O)(c1cccc(C2CC2)c1)N1CCCC(N2CC(C)C3(C2)CNC3)C1 N1(c2c(C)cnc(C)n2)CC2CCC(NC(c3cccnc3F)=O)CC2C1 N1(C(CC(C)n2ccnc2)=O)CC2CC2(CNC(C2CC(O)CN2C)=O)C1 N1(C(CCCC=C)=O)CC(NC(C2(C)CC3(CC3)C2)=O)CC12CCOCC2 C1(NC(C2(CCOC)CCN(C(=O)C(F)F)CC2)=O)CC2CCCCCC12 c1(-n2cc(CNC(C(C3CN(C(C)=O)C3)OC)=O)nn2)ccc(C)cc1F Cc1ccc(CNCC2CCCCN2C(=O)NCCCCl)nc1Br C1(CC(=O)NCCCN2C(C)CCC2)CCN(C(c2scnc2Cl)=O)C1(C)C CC(C)CC(C(=O)N1CCCCCC1C)NC(c1nnc(O)nc1O)=O Cc1ccc(C=CC(=O)NC(C)C(C)NC(c2ccc(Br)s2)=O)cc1C C(C1CCOCC1)=CC(=O)N(C)CC1CCCN1C(C1CCC1(F)F)=O c1(CC(=O)NCC2(O)CN(C(C3C(C)C3)=O)C2)ccc(Br)c(Cl)c1 C(CCCCn1cc(C2(Cl)CC2)nn1)NC(=O)NC1CCC1CF c1(CCCC(=O)OCc2cn(CCC(N3CCS(=O)CC3)=O)nn2)ccc(F)cc1 N1(C(C(C)SCC)=O)CCOCC(CNC(=O)C(C2CC(F)(F)C2)OC)C1 C1(C)(NC(C=CC(=O)OCC(C)C)=O)CCCN(C(=O)CC2CC2(Cl)Cl)C1 c1(C(=O)NC(C)C(CO)NC(=O)C(c2ccccc2)F)cc(Cl)ccc1O N1(C(Cc2c(C)ccs2)=O)CCCC(CCCCNC(C2OCC2(C)C)=O)C1 N1(C(C(C)N2CCC2)=O)CC2CCN(C(C3CCOC3c3ccncc3)=O)CC12 c1(C(=O)NCCC(C)N(C)C(C2C(F)(F)C23CC3)=O)cc2occc2s1 C1(COC)CC(CNC(c2csc(CO)n2)=O)N(C(=O)C(C)C)C1 c1(CCNCC(C)NC(=O)OC(C)(C)C)ccc(-n2cccn2)nc1 c1(C(N2CC3C(CNC(C(C)C(C)(C)C)=O)C3C2)=O)cccc2sncc12 c1(C(C2N(C(C(CC)C)=O)CSC2)=O)n[nH]c(C)c1Br.C(C)(C=O)OC(C)=O C(CCCC(C)NC(C1(F)CCCCC1)=O)NC(c1c(C)scc1)=O O=C(C1=C(Cl)CC1)NC1CCOC(C(=O)NCCC(CO)CO)C1 c1(C(N2CC(CNC(C(C3CCOCC3)C)=O)C(C)C2)=O)ccn(O)c(=O)c1 C=C=CCC(=O)NC(C1CCCCC1)C(=O)NC(C1CCOCC1)C C#Cc1ccnc(C(=O)NC2CN(C(=O)CNS(=O)(=O)N(C)C)C(C)(C)C2)c1 C1(NC(c2[nH]cc(C#N)c2)=O)CCC2CCN(C(c3ccc4cncn4c3)=O)C12 C(CCC(=O)NCCC(N1CC2(CC2)C1)=O)NC(C)=O c1(N2CC(COC)OC(C)(C)C2)nc(C)cc(=NC(C)c2ccc(Cl)c(F)c2)[nH]1 C1(C(N(CCCNC(=O)Cn2nccn2)CC)=O)CC(C(C)=O)C1(C)C N1(C(C(=O)NC(c2ccncc2Cl)C)=O)CCC(C)C(N)C1 c1(C(N2CCC(F)(CNC(c3n(C)ncc3)=O)CC2)=O)ccc2ncncc2c1 c1(N(C2CCCN(C(C3(C)CC(=C)C3)=O)C2)CCO)nc(OC)c(F)c(C)n1 C1(C(N(CCCC#N)CCCCN2CCOCC2)=O)CCC(C2(C(=O)OC)CCC2)O1 N1(C(C(C)OCOC)=O)CCCN(CCNC(=O)CCc2cscn2)CC1 c1(SC)ccc(N2CC(C(=O)NCC(C)NC(C3(C#N)CC3)=O)CC2=O)cc1 C1(C(=O)NC(C(=O)N(C(C)C)C)Cn2ccnn2)CC2CCC1C2 c1(C(=O)OC)ccc2c(c1)CCN(c1ncc(C)c(C)n1)C2C N1(C(=O)CCSCC2CCCCO2)CC(CNC(C2CC3(CCC3)C2)=O)C(O)C1 C(N=c1[nH]nc(C(c2ccco2)=O)s1)C1(C)CS(=O)(=O)C1 c1(NC(=O)CN2CCN(C(c3cc(F)cc(F)c3)=O)CC2)cc(CO)ccc1I CCC(CC)C(C)C(=O)NC1CC(F)(CNC(C23CCC(CC2)OC3)=O)C1 C1(C)(C(=O)OC)CCN(C(=O)NC(C)C)CC1 C1(NCC(=O)OCc2ccccc2)CCCC(Nc2nnc(S)s2)C1 C1(C(F)(F)F)(C(N(C2CCN(C(=O)C=CCn3cncn3)C2)C)=O)CCCCO1 C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(C(C)NC(C)=O)=O)C1 C(=O)(CCCCCCCCCO)N(C(C)CN(C(=O)C(Cl)=CCl)C)C c1(C(N(C2CN(C(C=CC=CCC)=O)CC2O)C)=O)ccc2ccc(Cl)cc2n1 CC1CCCC(C(N2CCOC(C(=O)Nc3ccnc(C4CC4)c3)CC2)=O)CC1 c1(CC)ccc(F)cc1C(N1CCNCC1C(=O)NC)C(=O)NC1CCC1 c1(CCC(=O)NC2(C)CCN(C(C(C=C=C)C)=O)C2)c(C)nc(O)nc1C C1(C(=O)N(CCC(=O)NCCN(S(C)(=O)=O)C)CCO)(OC)CCCCC1C CCCC(CCNC(=O)C(CCSC)NC(=O)C(C)N=[N+]=[N-])CCC N1(C(c2cn(C(C)C)nc2)=O)CCC(C(=O)NCCn2ccnn2)C1C c1(C(N2CCC(N(CCO)C(C3(C4CCC4)CC3)=O)CC2)=O)cc2c[nH]cnc-2n1 N1(C(c2c(C(C)C)nns2)=O)CCC2CN(C(C3CCSC3)=O)CC12 N1(CCOC)C2CCC1CN(c1nnc(-c3n[nH]cc3Cl)n1CC1CCOC1)C2 c1(C(=O)NC2C(NC(COC(C)C)=O)CCCC2)nn(C)c2c1CC(F)(F)CC2 N1(C(c2nnn3c2CCC3)=O)CC2CCN(C(=O)C(C3CCCCC3)F)CC2C1 c1(C(c2n(CCSC)nnn2)NCCc2nc(C)cs2)cncc2ccccc12 C1(NC(C(C)(C)C2CCOC2)=O)CCCCCC1NC(=O)Cc1csnn1 C(=O)(C1=CCCOCC1)N1CC(C)(C)C(NC(=O)CCc2ccc(Br)s2)C1 Cc1nc2sccn2c1C(=O)NC1CC12CCN(C(C1CC1C1CC1C)=O)CC2 CCC(CC)(C(=O)N1CC2CN(S(=O)(=O)c3nccs3)C2C1)C(=O)O C1(C(=O)NCCCNC(c2ccc(CO)o2)=O)CC2CCC1C2 c1(C(N2CCC(CCNC(c3nc(C4CC4)cs3)=O)C2)=O)ccc(O)cc1 C1(C(=O)NCc2c(C)nccc2)CC2(C1)CN(C(c1ccc(O)c(F)c1)=O)C2 Cc1ccc([N+](=O)[O-])c(CC(=O)NCCCN(C)C(c2c(N)sc(C)c2C)=O)c1 N1(C(C=CC)=O)CCCC2CN(c3ncc(C#N)cc3Cl)CCC12 N1(C(c2cc3cccnc3[nH]2)=O)CCC2CCN(C(C3(C(F)F)CC3)=O)CC12 C(=O)(CC1OCc2ccccc21)NCC(C)(C1CC1)NC(=O)C1=CCS(=O)(=O)C1 C#Cc1ccc(C(=O)NC2CN(C(c3ccc(SC)s3)=O)CCC2C)nc1 C1(C(=O)NCC2(O)CCN(C(c3nc(C)sc3C)=O)C2)CCOC(=O)CC1 N1(C(c2scc(C#N)c2)=O)CC2CC1CN2C(c1cn(CC(F)(F)F)cn1)=O C1(CN(C(CCC)=O)CC)CCCC(NC(C2(n3ccnn3)CC2)=O)C1 c1(-c2ccc(CC)nc2)cccc2[nH]nc(C(=O)NCc3ccc(CO)cn3)c12 C1(NC(=O)COCC(F)(F)F)CCCN(C(C2CCN3CCCC3C2)=O)CC1 CC#CCCCC(=O)NCC1(OC)CCN(C(=O)CC(=O)OCC)C1 N1(C(c2c(CNC(=O)CC3CC34CC4)nccc2)=O)C2CCCC1COC2 C1(c2ccc(OC)cc2C)NC(=O)N(CCc2nccs2)C2=C1C(=O)NCC2 N1(C(N(C)Cc2ccccc2)=O)CCC2CCNC(=O)C2C1 c1(-c2cn(CC(CCOC)NC(=O)CC3CCC3)nn2)ccc(F)c(C(C)=O)c1 Cc1ccc(NC(C2(F)CCN(C(c3sc(N(C)C)nc3C)=O)C2)=O)c(SC)n1 C1(CNC(c2c(C)ccn2C)=O)C(O)C(O)CN1C(c1occc1F)=O c1(CNC(C2(C=C)CCC2)=O)nc2c(s1)CN(C(=O)CCc1ccsc1Cl)CC2 O=C(CCCC1CCC1)NCC(=O)NC(c1ccccc1)CO C12(CNC(C3CCC3)=O)CCC(C1)N(C(=O)Cn1ncc(Br)n1)C2 C1(C2CN(C(C3(C)CC=CCO3)=O)C2)(NC(CC=C(C)C)=O)CC1 N1(C(CCOC)=O)CC(C)N(C(C2CCCC(C)C2)=O)CC1C N1(C(C(C)(C)SC)=O)CC2(NC(c3cc(N)c(F)cn3)=O)CCC1CC2 CC(CC(=O)NC1CC(O)(CNC(c2cc(C(N)=O)co2)=O)C1)n1cccn1 C1(C)(C(c2nnnn2Cc2nnn(C)n2)(C)NC(COC(C)C)C)CCCCO1 CCC(COC)C(=O)NCCCC(=O)Nc1cnn(C(F)F)c1 O=NN1CCCC1C(=O)NCCN1CCN(C(C2CCCCNC2)=O)CC1 N1(C(C2N(CC)CC2)=O)CC2CC1C2CNC(=O)CCC(C)N(C)C c1(C(=O)NC(C(C)(C)C)CNC(c2cccc(O)n2)=O)cc2sccc2n1C c1(C(C)C(=O)NC2CCC2NC(=O)Cc2cnsc2)ccccc1S(N)(=O)=O C1(CCC)(NC(c2cn(C)cc2C)=O)CCN(C(c2cnnn2CC)=O)CC1 C1(OC)CCN(C(=O)CSCCNC(c2ccnc(CO)c2)=O)CC1C C1(CNC(C(C)(C)NC(=O)C=CCO)=O)CCC2(CC2)C1 N1(C(CCN(CC(F)(F)F)C)=O)CCC(CO)(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(=O)NC(CNC(C2(C)CC2)=O)C2CC2)cccc(OCC)c1.C(C)(C)(C)OCCF CC1CC(C(=O)N2CCCC(NC(=O)CCCCO)C2C)=NO1 c1(C(N(CC#C)C(C)C)=O)coc2c1CN(C(=O)C(C(C)C)SC)C2 c1(NC(c2ccccc2)C(N2CCCC(C#C)C2)=O)ccc2oc(C)nc2c1 C1(C)(C(=O)NCCN(C)C(c2ccnc(-c3cc[nH]n3)c2)=O)CC2CCC1C2 n1(CC(=O)NCC(C)NC(C(c2c(C)n[nH]c2C)C)=O)ccc2c(N)cccc12 Cc1ncc(Br)c(C(=O)NCCN2CCN(C(=O)CC3CCCCCC3)CC2)n1 C1(NC(c2c(C)nccc2)=O)CC(N(C)C)C12CCC2 c1(C(N(CC(c2ccccc2)NC)C(C)C)=O)c(Cl)cc(Cl)nc1C c1(OC)cc(CCC(=O)NC2CC(C)N(C(c3ccc(CO)nc3)=O)C2)nn1C C(=O)(CCCC(=O)NCC1CN(C)CCN1C(c1ccc(Cl)o1)=O)OC c1(C(=O)OC)cc(NCCCNCCc2ncc[nH]2)cc(Br)c1[N+](=O)[O-] c1(CCC(=O)OC)cc(NC(c2nc(CSC3CC3)oc2C)=O)c(C)o1 CCCC(C)(CC)C(=O)NC1COCC1NC(=O)Cc1c[nH]c(=N)nc1O N1(C(c2c(CC)nco2)=O)CC(OC)C(NC(c2ccccc2OC(C)C)=O)C1 C1(C(=O)NCC2(CCC=C)CC2)CC(NC(=O)CN(C)CC)CCO1 c1(C(N2CC(OC)C(NC(=O)C(F)C3CCC3)C2)=O)nnn2c1C(=O)NCC2 c1(C(=O)NC(CNC(c2cnc(OCC)s2)=O)(C)C2CCC2)cc(O)nc(O)n1 C(=O)(C(F)C(C)C)NC(CC)COc1ccccc1 C(C(=O)NCCOCCN(C(=O)CCC1CC1(C)C)C)(C1CC1)SC C1(NC(c2c(C)nco2)=O)CN(C(=O)C2=C(Cl)CCOC2)C2(CCCCC2)C1 C1(C)(NC(c2nccc(CC)c2)=O)CCCCC1C(=O)Nc1cnn(CCOC)c1 N1(C(CC(C)c2cnn(C)c2)=O)CCC2CN(C(=O)CC3CCC3)CC2C1 N1(CC)CC2(C)CN(Cc3ccccc3)CC2(C)C1.c12cccn1NC(=O)NC2 c1(C(=O)NCC(C)(C)CC(C2CCCC2)OC)cc(Cl)c2n[nH]cc2c1 c1(C(N2C(C(=O)Nc3cc(OCC)c(C)cc3)CC2)=O)cc2sc(F)cc2[nH]1 CC(CC(=O)N(C)CC1CCN(C(C2CC(O)CN2C(N)=O)=O)CC1)P(C)(C)=O CCC(CC(C)C)C(=O)N1CCC(C2CCCN2C(C2(CO)CCCC2)=O)CC1 C12(CNC(C3C(CC)C3)=O)CCCCC1N(C(=O)C(C)CCOCC#N)CCC2 Cn1cnc(C(=O)NC2(CNC(=O)Cc3cnns3)CCC2)n1 c1(CNC(C2CCCN(C(=O)Cc3cccs3)CC2)=O)cccc2occc12 C12(C3CNC(=O)N3)CCC(CC1)C2.Cc1cnn(CC2(O)CCSC2)c1 Cc1nn(CC(C)C)c(C)c1CN1CCN(C(=O)NC(C)(C)C)CC1C(F)(F)F c1(C(N(C2CCN(C(=O)C(C)(C)CCl)C2)C)=O)cc([N+](=O)[O-])ccc1Br CC1CC(C(=O)N2CCC(OCC(=O)NC(C)CC(N)=O)C2)=NO1 CCCC(C)(O)CC(=O)N1CCOC(CN(C(=O)Cc2occc2C)C)C1 c1(C(N(C)CC2CCN(C(=O)CCC3CC3)C2)=O)ccc(F)c2ccncc12 C12(C(N(CCCSc3ccc(C(N(C)CC)=O)cc3)C)=O)CCC(O)(CC1)CC2 N1(C(C2(O)CC(C)(C)C2)=O)CC2CC1CC2NC(=O)CO Cc1nocc1C(=O)OCC(=O)NC(C(C)(C)C)c1cccs1 C(=O)(CC(C)CC(C)C)N1CCC(c2cn(CC(CC)(C)C)nn2)CC1 c1(C(=O)NC2C(NC(c3cnn(CCC)c3C)=O)CCC2)ccc(C#N)cc1C c1(CN(CCCOCCC(=O)NCC)C)cc2cc(F)ccc2[nH]1.CC(=O)N1CC12CNC2 C1(C(=O)NC2(C(=O)NC3C(C)CCC3C)CC2(C)C)CC(=O)OC1(C)C CC1CN(C(=O)CCSCC#N)CCCN1C(c1ccc(OC(F)(F)F)nc1)=O c1(OC)cc(C(=O)Nc2cccc(F)c2Cl)c(NCc2cc(Cl)cnc2C)cn1 N1(C(C2CC3CCN(C(CC(=O)NC)=O)CC32)=O)CC2(C1)CN(C)CCO2 CC1CC(C(=O)NC(C)(C)CF)CN(C(=O)Cc2ccnc(O)c2)C1 CC1(C)CCN(C(c2nc[nH]n2)=O)C1C(=O)NC1CCCC1N=[N+]=[N-] Cc1ccc(N(S(=O)(=O)C(C)C)CC2CCOC2)c(C)c1 Cn1cc(C=CC(=O)NC2(C)CC(NC(C3(CC(F)F)CCC3)=O)C2)cn1 N1(C(C2N(C(CC)=O)CSC2)=O)CCCC(NC(=O)C=C(C)C2CC2)C1 C(=O)(C(C(C)C)OC)NCCCCN(C(C(c1cncnc1)OC)=O)C C=CC(C)(CC)C(=O)N1CCC(CO)C(NC(c2cc(C3CC3)ncn2)=O)C1 C=CC(CCC)CC(=O)NCC(CCOC)NC(c1c(F)cc(Cl)cc1F)=O CC(O)(Cc1ccccc1)C(=O)NCCC(O)CNC(c1coc(C(F)F)c1)=O N1(C(c2cccc(COC)c2)=O)CCN(C(=O)C#CC(C)C)CC1CC(F)(F)F C1(N(C(=O)Cn2cnc(Br)c2)C)CN(C(=O)Cc2cccs2)CC12CC2 Cc1ccc(F)c(OCC(N2CCC3(NC(=O)CSC4CCC4)CC3C2)=O)c1 CC1(C)CN(C(=O)C=CCF)CC1C(=O)NCC12CCCCC1C2 c1(C(C(=O)N(C(CN(C(COCCC=C)=O)C)C)C)C)ccc(Br)cc1 c1(NC(c2scc(C)n2)C)nc[nH]c(=NCc2ccc(F)c3cc[nH]c23)c1C Cc1cn2c(C(=O)NCC3CCN(C(C4CCCS(=O)(=O)C4)=O)C3)c(C)nc2s1 CC(=O)CCCC(=O)N1CCC(C)C1CNC(c1ccc(C(C)C)nc1)=O NS(=O)(=O)C1CC(C(N2CCC(NC(=O)CC3CC(F)C3)CC2)=O)C1 C=C(Cl)CCC(=O)NC1CN(C(=O)C(C2CCCC2)N(C)C)CC1CC1CC1 C(=O)(CCC(CF)CF)NC1C(C(N2C(C(=O)NC)CC(O)C2)=O)COCC1 C#Cc1ccccc1CNC(=O)CC(C(C)C)NC(C)=O.C12CCN(C1)C2=O NC12CCOCC1CN(C(=O)C=CCN1CCOCC1)C2 C1(C)(NC(c2nc(CC(C)C)sc2)=O)CCN(C(=O)C(C)CN(C)C)C1 N1(C(c2ccc(C)nc2)=O)CC(C(=O)NCC2(C#N)CC2)OC(C)C1 C12(CNC(C(C)NC3CCCO3)=O)CC(NC(c3ccco3)=O)(CCO1)C2 C1(C(N(C2CC(SC)C2)C)=O)C2CC1N(C(c1ccc(CO)s1)=O)C2 CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC2CCN(C)C2)C1 c1(C(N2C(CNC(C3N(C(C)=O)CCCC3)=O)C=CC2)=O)nccc2n[nH]cc12 N1(C(C(C)=C2CCC2)=O)CCC(F)CC1C(=O)N(CC(C)(F)F)C N12CCN(CC1)C2=O.C(C(O)C(=O)NCC1CCC1)OC S(=O)(=O)(c1cccnc1N)N(C1CC(O)C1)C.Cc1nnsc1CN C(=O)(C1=CC2(CCOC2)C1)NC1COCCN(C(Cc2scc(C)n2)=O)C1 Cc1cccn2cc(C(=O)NCC(CO)NC(=O)C(CO)C(C)(C)C)nc12 CCCCCCCC(F)C(=O)N1CCN(C(C2COc3ccccc3C2)=O)CC1 C1(NC(c2nc(C)oc2)=O)CN(C(c2cnsc2)=O)CCC1C C(=O)(C(C)(CC)C(N)=O)NCC1CCCCN(C(C(F)=CC)=O)C1 C(C)(C)(C(C)CC(=O)N1CCSCC1)NC(c1nc(C)oc1)=O C1(C(NOC(C=C)C)=O)CC(C)CN(C(C2CCC2COCC)=O)C1 c1(C(=O)NC(CC)CNC(=O)C(c2ccccc2)SC)ccc2cnccc2n1 C(CC(C)(C)C)(C(=O)N1CCCC(NC(=O)OC)C1)NC(c1cncc(NC)c1)=O c1(CC(N2CCC(CCNC(c3ccccn3)=O)CC2)=O)ccc2nc[nH]c2c1 c1(N(CCCCOC)C)cccc(S(=O)(=O)NC2CCS(=O)(=O)C(C)C2)n1 CC(C)CCC(=O)NC(C(N1CCC1(C)C)=O)c1ccoc1 c1(OC)ccc(CCC(=O)N(N(C=O)CC(C)OC)C2CC2)cc1OC C12(C(=O)NC(C)C(N)=O)CCC(n3cc(-c4cccnc4)nn3)C1C2 C(=O)(CCC(=O)NN(C)C)N(CCCCCCNC(CC(C(C)C)C)=O)C C1(CNC(CC2(COC)CCOCC2)=O)CCCCN(C(=O)CCC(N)=O)C1 CN1CCC(C(=O)NCCC2(O)CN(C(c3[nH]ccc3-c3ccccc3)=O)C2)C1 c1(C(N)=O)ccc(CCC(N2CCCC2c2cccc(Br)c2)=O)cc1 C1(NC(c2ccc(C(N)=O)cn2)=O)COC2(CNC(C3CCCO3)=O)CC1C2 c1(CC)c(C(=O)NCCCCNC(=O)CCN2CCNC(=O)C2)nnn1CC N1(C(c2c(CC)ocn2)=O)CCC(NCCNC(=O)C2=CCSC2)CC1C Cc1nc(NC2CN(C(C3CCOC(C(C)C)C3)=O)CC2C)ncc1[N+](=O)[O-] C=C(Cl)CC(C(=O)N(C(CSCC)CC)C)NC(=O)CC1CCC(C)(C)O1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CCC(NC(CCSCCC)=O)CC1 c1(CC(N2CCC(N(C(C=CC)=O)C)C2)=O)ccc(OC)cn1 C12(C(=O)OC(C)(C)C)CCC(C(=O)N(C3(C4CCCO4)CC3)CCO)(CC1)O2 c1(CNCC(CCC=C)O)cc(C(=O)OC(C)=O)ccc1C C(=O)(C1CCc2nnc(C)n21)NCCC1N(C(Cc2cc(C)no2)=O)CCSC1 c1(CC=C(C)C)cccc(C(=O)N(CCCCCNC(C2CNC(=O)O2)=O)C)c1 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(CNC(CCC(CC)OC)=O)C N1(Cc2cc(C(=O)OC)n[nH]2)CCC2C(C1)NC(=O)CCN2C C(CNC(C1COC(C)(C)C1)=O)(CC)(CC)NC(c1nc(CCC)oc1)=O C1(CC(=O)OC)COC(C)(C)CN1C(=O)Oc1ccc(OOC(C)(C)C)c(C)c1.O c1(C(N2CC(C)(CNC(C(CC)O)=O)OCC2)=O)cc2c(nnn2C)s1 C#Cc1cccc(CC(=O)NC(C)C(C)(C)NC(=O)CCCN(C)C(C)C)c1 C(=O)(CC(C)C(C)(C)C)N1CC(NC(C(C(C)(C)O)OC)=O)C(C)CC1 C(=O)(C1=NOC(C)C1C)NC1C2N(C(c3c(OC)cccc3)=O)C(CC2)C1 N1(C(CCC)=O)CCCC(C(N2CCCC2COC)=O)C1CC C=CC(C)CC(=O)NC(CCOC)C(=O)NC1CCCC1CCOC c1(CN2C(C(=O)Nc3ccc(C(F)(F)F)nc3F)CCC2)c(O)cc(F)cc1F C1(C(N2CC(OCCOC)C2)=O)CC12CCN(C(c1ccsc1C)=O)CC2 C1(C(=O)NCC(C)CC2CCC2)CCC(C2CC2)N1C(=O)Cn1cnnn1 CCCCC(C(=O)NC)NC(=O)C(CC)N(CC(N1CCCC1)C)CCOC CC1CC(C(=O)NCC2CN(C(c3cc(-c4cccn4C)[nH]n3)=O)CCO2)=NO1 C12(C(=O)NC3CC(C(C)NC(=O)COC4CCOCC4)C3)CC(C)(C1)OC21CCC1 N12CC(CCC1C)NC(=O)c1ccc(cc1)C2C.Cc1ccccc1CO N12CCC(F)(C1)C(=O)NCC1(CC1)C2=O.C1(SC)(CF)CC1 C1(CC#C)(C(=O)NCC2CCCC2(C)C)CCN(C(c2ccc(CC)nc2)=O)C1 c1(CNC2C(C(=O)Nc3c(C)cnn3C(C)C)CCC2)ccc2ncnn2c1 N1(C(C(CC)n2ccnc2)=O)CCC(C)(CNC(c2c(C)ncn2C)=O)C1 c1(CNC(C(=O)NC(C2CCOC2)CC)=O)cc(OC)c(OC)cc1OC N1(C(c2ccccc2)C)CCC(C)(Cc2cccc(Br)c2)C1.c12cn(nn1)C2 CC(C)(C(=O)NC1CCCC(CNC(=O)C=CCCc2ccccc2)C1)C(F)F C(=O)(C(C)(C)CCCO)NC1(CC=C)CN(C(c2coc(C(F)F)c2)=O)C1 c1(OCC)cc(C(=O)NCC(C)CNC(c2cncc(OC)c2)=O)ccc1C c1(C(=O)NCC(C)CN(C(=O)C(C)C2CCCC2)C)ccc(-c2nc[nH]n2)nc1 C1(C(=O)NC2CC(C)N(C(C34CC5CC3C4C5O)=O)CC2)CNC(=O)CC1(C)C c1(SC)ncc(N)c(C(=O)NCCCCNC(c2cc(F)cnc2O)=O)n1 C(=O)(N=c1cc(CO)[nH][nH]1)c1cnc(NC(C2CCC3(CC2)COC3)=O)c(O)c1 CC(C)CC(=O)C(=O)NC1CC(OCC(N2CCC(C(C)C)C2)=O)C1 C1(C(N2CC(OCCNC(C3CC4(CCC4)C3)=O)C2)=O)CCCC(C2CC2)O1 C(N=c1ccnc(NCCC2CCCCC23CC3)[nH]1)c1occ(C)n1 C(=O)(CC(C)(O)C(F)(F)F)NCC1(NC(C2(c3n(C)ncc3)CC2)=O)CCCC1 c1(C(=O)NC(C2(O)CN(C(C3CCCC3F)=O)C2)C)ccc(Br)s1 c1(OCC)ccc(C(=O)NC(c2ccnc(F)c2)C(=O)O)cc1 c1(C(=O)OCC)ccccc1C(C)C.C12(CC1)CNC(=O)N2.OCC O=C(CC(C(F)F)n1ccnc1)NCCN(C(=O)COC1CC=CC1)C1CC1 C1(C(=O)NCC2CCC23CCC3)CCC2(CC2)N1C(=O)CN1CCSCC1 N1(C(C2C(C)(C)C2)=O)C2CCC1CN(C(=O)C#CC1CCC1)C2 Cc1cc(C(=O)NCC2COC(CNC(=O)C3=NOC(C)C3)C2)c(C)n1C1CC1 C1(CC=C)(NC(=O)CSC)CCN(C(c2ccc(NCC(C)(C)C)cc2)=O)CC1 C1(C(N2CC(C(=O)NCC(=O)N(C)CC)(COC)C2)=O)CC2CC(=O)C1O2 C(=O)(C#CC1(C)CCCO1)N1CCC2(CC(C(N(CC(F)F)C)=O)C2)C1 c1(C(=O)NC2C(C(N)=O)C2)ccc(-c2cncnc2)cc1.c12cc([nH]n1)N2 c1(NC(CCCCC)C2CC2)nc2ccccc2nc1NCCOC1CCCO1 C1(C(N2CC(OC)C(NC(c3cnc(SC)s3)=O)C2)=O)CC(S(C)(=O)=O)C1 C1(NC(C(CO)NC(C(C)C)=O)=O)CCCCN(C(c2ccncc2N)=O)C1 c1(OCC)cccc(NC(C2CC(F)CN2C(C2CC2C(C)(C)C)=O)=O)c1 c1(C(=O)NCCCC(C)NC(=O)C(C)N(C)C)ncnc2c1cnn2C c1(C(N(C2CN(C(c3c(CC)csc3)=O)CC2(C)C)C)=O)cccn2nnnc12 C1(C(=O)NCCc2ncn(C)n2)CC(NC(=O)CN2CCC(=O)CC2)CCO1 c1(C(=O)NC(CN(C(=O)CC2CC3CC3C2)C)(C)C)ccc(S(N)(=O)=O)s1 C1(NC(CSc2ccc(OC)cc2)=O)CN(C(=O)CC2CCN(C)C2)CCC1F Cc1ccc(CC(=O)NCC2CC2NC(c2cn(C(C)(C)C)nc2C)=O)c(C)c1 c1(N2CC3CC(C)CN3CC2)nc(C(F)(F)C(F)(F)F)nc(=NCCCN(C)C)[nH]1 C1(c2nnnn2C2(C)CC2)(NC(c2cccc(CC)c2)(C)C)CCOCCC1C c1(CC(C2CC2)NC(=O)NC2CCCCC2)ccccc1 CC(C(=O)NC1(C)CC(NC(=O)CCOc2ccc(F)c(F)c2)C1)S(N)(=O)=O CCCC(C)(CC)C(=O)NCC(C)(C)CNC(c1ccc(=O)n(CC(C)O)c1)=O N1(CC)CC(NC(=O)C(c2ccco2)NC(c2cc(C(F)F)[nH]n2)=O)CCC1=O C#Cc1cncc(C(=O)NCC2CCC(C(=O)NC(c3nc(C)cs3)C)O2)c1 C1(CNC(c2c(C)cno2)=O)CCN(C(c2cc(Cl)nn2C)=O)C1(C)C N1(C(C(COCC)(C)C)=O)CCC2CN(C(=O)C=C(C)COC(C)=O)CC2CC1 c1(C(C)=O)ccc(CC(=O)NC2CCC2CCNC(=O)C(=O)N(C)C)cc1 n1(CC)cnc2[nH]c(=NC3CCS(=O)CC3)nc(N(CCCCOC)C)c12 C1(NC(C(C)NC(N)=O)=O)CCC(CNC(=O)CCCn2ccnn2)CC1 C(C(=O)NCc1ncoc1C1CCN(C(c2cnoc2C)=O)C1)(C(C)(C)C)OC c1(C(=O)NC2C(NC(C=CCC)=O)CCC2)ccc(C)c(C(=O)OC)c1 c1(C(C)C)n[nH]cc1C(=O)NC1COCC1C(=O)N(C)Cc1ccon1 CCC(CC(F)F)C(=O)N1CCOCC(NC(=O)CCC2(C)CCC(=O)N2)C1 C1(NC(c2c(C)nc(CO)s2)=O)COC2(CCN(C(c3ncn(C)c3C)=O)C2)C1 C(CCCCCCCc1ccccc1)(c1nnnn1C(C)C)NCCC(CC)(C)C C(c1cccc(C)c1)=CC(=O)N(CCNC(=O)CCC1CC1(C)C)CC N1(CC)CCN(CCC(=O)NCC#CCNC(=O)CC2CCCO2)CC1 C(C)(C)(C(=O)NCCCCCNC(C1CC(O)C1)=O)OCC C1(C(N(C2C(C)C2C#N)Cc2c(OC)n(C)nc2)=O)CC(C)CCN1C(=O)CC#N c1(NC(c2ccc(NS(=O)(=O)C(F)(F)F)cn2)=O)cc(Cl)nc(Cl)c1Cl c1(C(N2CCCC(CNC(CCCC)=O)C2)=O)ccn2c(O)nnc2c1 C1(C(N(C)Cc2cn(CC)nn2)=O)(NC(c2cn(C)c(=O)cn2)=O)CCCC1C CCC(C)C(CC(=O)NC1CCC(=O)NC1(C)C)NC(=O)C(C(C)C)N(C)C C1(C)(C(=O)NCC(CNC(CC2CC(OCC)C2)=O)C)CC2(C1)CC(F)(F)C2 N1(c2c(Cl)cnc(OC)n2)CC2(CCCC2NC(=O)C2=CC(C)(C)C2)C1 N1(C(CCOC(CC(C)C)C)=O)CCCC(N(C)C(C2(O)CCOCC2)=O)CC1 CCCCC(CNC(=O)Cc1sc(SC(F)F)nc1C)NC(=O)CCCOC C1(NC(c2cc(C)sc2)=O)CN(C(C2CC(C)CC(C)C2)=O)C(C)(C)C1 Cc1cc(C(=O)NC2(CNC(=O)CSc3cn[nH]c3)CC2)c(C)n1CC(F)(F)F c1(C(=O)NC23CC(NC(c4c(CC)cco4)=O)(C2)C3)cc(Cl)cnn1 N1(CC(=O)NCCNC(CC(CC)C2CCC2)=O)CCC(C)(C)CC1 C1(C(C)C#N)CCN(C(C2C3CN(Cc4cc(Cl)ccn4)CC23)=O)CC1 C1(C(C)(C)NC(C=C(CCC)C)=O)CCN(C(=O)CCC(C)N(C)C)CC1 C1(c2ccc(OC)cc2)CN(C(=O)COC)CCN1C(=O)CC1CC2CC1C2 C#CCC(O)C(=O)NCCCOCCN(C)C(c1n[nH]c(C)c1Br)=O N12CCCCC1C2=O.c1(CCCN2C(CNC(N)=O)CCC2)ccc(F)cc1 C1(C(=O)NCCCNC(C2CC2(C)C(F)F)=O)(CC)CCCC1 Cc1cc(C(N2CC(NC(c3c(C)ncn3C)=O)CC(C)C2)=O)ncc1N N1(C(c2cc(C)n(C)n2)=O)C2CCCC1CN(C(=O)C(F)CC1CCOC1)C2 c1(C(=O)NC2(COC)CN(C(C3CCC(C)O3)=O)C2)ccc2nnc(S)n2c1 C(CO)(CC(C)(C)C)NC(c1ncn(CCNC(c2cc(COC)[nH]n2)=O)c1)=O N1(C(c2c(CCC)[nH]cc2)=O)CCC(C(=O)NC(C(N)=O)C2CCCC2)C(O)C1 c1(C(N2CCC2CNC(C2C(=O)NCCC2C)=O)C)cccc2ccccc12 N1(C(c2cc(C)no2)=O)CCC2(CC1)CCN2C(c1cc(Br)c(C)cc1O)=O C#CCC(C)(CC)C(=O)NCC(C)(C)C#CC(=O)Nc1ccc(F)nc1 Cn1nc(Br)cc1C=CC(=O)NCC(O)CNC(c1cc(Cl)ns1)=O CC1SCCCC1C(=O)NCCN(C)C(c1cc(-c2ccn(C)n2)on1)=O c1(C(N2CCC3CN(C(C4C5CCCOC45)=O)C3C2)=O)cccc2nc(Cl)cn12 C(=O)(CC(C)(C)CC(=O)OC)N1C2CC(NC(C(CCC)NC(N)=O)=O)C1CC2 c12cc(O)ccc1C(=O)N2.N1(C(C=CC(=O)NC2CC(OC)C2)=O)CCCCC1 C1(N(C(C2CC2c2ccsc2)=O)CC=Cc2ccccc2)CC2(CCNCC2)C1 CCCCS(=O)(=O)CC(=O)NC1CCCC(NC(c2nc(C)c(N)cc2C)=O)C1 C1(CNC(CC=CCC)=O)CN(C(=O)COc2cc(C)on2)CC1(F)F C(C1(C)COc2ccccc21)NC(NNC(c1ccc(OC(C)C)cc1)=O)=O C(c1ccncc1)=C(C)C(N1CC2C(CC(N3CC(N4CCCC4)C3)=O)C2C1)=O C1(CNC(CCCNC(C)=O)=O)CCN(C(c2cc(C(F)F)nn2C)=O)CC1C C(=O)(C1CCc2cc(C)ccc21)N1CCN(C(C2=C(C)CC2)=O)CC1C C#CCC(C)(CC)C(=O)NC(C)CCNC(c1ncc(C(C)C)s1)=O C(=O)(CC(C)(C)CC=C)NCC1(C(=O)NCC=C)CC12CCC2 c1(C(=O)NC2CC(NC(COc3cccc(C)c3)=O)C2)cn(C)c(=O)nc1O C(=O)(CCC1(NC(=O)CCC2CC2(C)C)CCC1)N(C1(CC(F)F)CC1)C C1(NC(COC(C)=O)=O)CCCC12CCN(C(c1cccc3nsnc13)=O)CC2 N1(Cc2c(C)ccnc2)CC2CCC(C1)C2NC(=O)C(C)C C(=O)(C1=NNC(C(F)(F)F)C1)NCC1C2CN(C(c3nn(C)c(Cl)c3)=O)CC21 c1(CC)cc(C(=O)NN2CC(C(=O)NC3COCC3N(C)C)(CC)C2)ncn1 Cc1ccccc1C(C)CC(=O)NCC1CCCN1C(=O)C(C(C)C)NC(N)=O N1(C(c2cc3c(o2)CCCC3)=O)CCC(N=c2ccc3nncn3[nH]2)CC1 CN1C(=O)CSC1=CC(=O)NCCCN1CCN(C(C2CC3CCC2O3)=O)CC1 CCCC(CC)CCC(=O)N1CCOC(C(=O)NCCCCCCF)CC1 c1(C(N2CCC(C)(CCNC(CNS(C)(=O)=O)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(CC(=O)NC(CN(C(CCOCCC)=O)CC)(C)C)ccnc(OCC)c1 c1(C(N(C(c2cccc(Cl)c2Cl)C(=O)NC(C)C)C)C)cccc2ccccc12 N1(C(C2(COC)CCOC2)=O)CCC2CCC(C1)N2C(C1CC(O)C1)=O c1(OC)ccc(CN2CCCC2CC(=O)Nc2cnc(O)c(C)c2)c(OC)c1 c1(C(=O)NC(C(CC)C)C(=O)N2CCN(C(=O)CO)CC2)cc2cccnn2n1 N1(C(CCC2CCN(C(CC(C(C)C)O)=O)CC2)=O)CC(=O)NC(C)(C)C1 n1(CCC)cc(Cl)c(C(=O)NCCC(C)CCNC(c2cnn(CCC)c2)=O)n1 C1(c2cccc(F)c2)(NC(C(C)=CC)=O)CCN(C(=O)CC(C)(C)C)C1 C1(NC(c2c(C)c[nH]c2)=O)CC(O)CN(C(c2cn(C)nc2-c2ccoc2)=O)C1 c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CCCC2)c(Br)nc2n1CCC2 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC(NC(c2cnc(OC)s2)=O)C2(CC2)C1 C(CCC(C)CC(=O)NC1CN(C(c2cccc(C)c2O)=O)CC1(F)F)=C(C)C C(C1CCCn2ccnc21)NC(COc1cccc(C(C)(C)C)c1)=O c1(C(n2cc(-c3ccc(Br)s3)nn2)COC)ccccn1 c1(C(N2C(C(C)(C)NC(=O)CC3CC=CCC3)CCC2)=O)ncncc1Cl N1(C(C(C(=C)C)(C)O)=O)CCCN(C)CC1c1ccc(C(=O)OCC)cc1 c1(C(N2C(C)C(C)N(C(=O)CCN3CCC3)CC2)=O)nc2c(s1)CN(C)CC2 C=CCC(CC(C)C)C(=O)Nc1ccccc1OCc1cccs1 c1(C(=O)NCC2(C)CN(C(C3CCS(=O)CC3)=O)CCO2)cnc2[nH]ccc2n1 Cc1cc(C)n(CCC(=O)NCC2CN(C(=O)CC3NC(=O)NC3=O)CC2C)n1 CC1CC(=O)NCCOCCN(C)C1=O.c1(SCC(=O)NC2CC2)ccccn1 c1(C(=O)NC(CN(C(=O)C(C)c2cc[nH]n2)CC)C)cc(F)ccc1NC Cc1cc(F)c(NCCn2cnc(C)c2C)c([N+](=O)[O-])c1 Cc1ccc(OCC(=O)NC2C=CCN(C(=O)C(C3CCCCCC3)O)C2)c(C)c1 N1(C(c2ccn(C)c2)=O)CC2=C(C1)CN(C(C1CCc3ncsc3C1)=O)C2 CC1CC(=O)NC(C(N2CCCC(CC(=O)NCC3CNC(=O)C3)C2)=O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(CC1CN(C(CC2CC(OCC)C2)=O)C1)C c1(C(=O)NCCN2CCN(CC3CC3)CC2)nc2cc3ccccc3cc2[nH]1 c1(C(=O)NCCC(C)N(C)C(C23CCC(CC2)C3)=O)cc(N)cc(S(C)(=O)=O)c1 N1(C(C2CC(O)(CNC(C=CC)=O)C2)=O)CCCCCCC1CC c1(OC)ccc(NC(C2CC2NCC2(Br)CC2)=O)c(Br)c1 C1(C(=O)NCC2CC(O)(CNC(COCC(C)C)=O)C2)CCCCN1S(C)(=O)=O C1(CC=CC(=O)NC(C2CCOC2)C#C)(NC(=O)C(C)N=[N+]=[N-])CCCCC1 c1(CN(CCOC)CC2(Cc3ccc(F)cc3)CC2)ccnc(F)c1 c1(C(=O)NCC=CCCNc2cc(OCC)ncn2)cc2sccc2[nH]1 c1(C(=O)NC(C(C)NC(=O)C(C2CCOCC2)O)CO)c[nH]c(=N)c2[nH]ccc12 Cc1sc(C(=O)NC2(C)CC(NC(c3c(Cl)ccc(Cl)c3O)=O)C2)cc1[N+](=O)[O-] O=C(C1=CNC2=NCCCN12)N1CC2(CC(NC(C3(C4CC4)CCC3)=O)C2)C1 c1(C2(NC(=O)NC(C#N)C(N)=O)CC2)ccc(C(F)F)cc1 c1(C(=O)NCC2N(CC#CC)CC2)sc(Cl)nc1C N1(c2snc(C)n2)CCCC2(CCN(C(=O)C3CCCc4c3ncn4C)C2)C1 C(=O)(CCCN(C(=O)C(C)CN(C)C)C)NCCCOCCOC N1(C(=O)Cc2ccc(O)cc2)CCCC2(C1)CN(C(c1cnn[nH]1)=O)C2 CCCCC(CC)CC(=O)NC1CC(CC(=O)NCCOCC)C1(C)C N1(C(=O)NC(C#C)C)CCC(C(C)(C)Cc2ccc(C(C)(C)C)cc2)CC1 C(=O)(CCCC(=O)N(C1CN(C(C2CC(F)(CO)C2)=O)CC12CC2)C)OCC C1(C(=O)OCc2snc(C)n2)CCCCN(C(=O)OC(C)(C)C)C1 N1(C(c2c(CC)cc(C)cc2)=O)CCC2CN(C(c3cc(Cl)nn3C)=O)CC12 CN1CCC2(CC1)CC2C(N1CCC(O)(NC(=O)Nc2ccccc2)CC1)=O Cc1ccnc2nc(C(=O)NCCC3CCN(C(=O)CC4CCOC4)CC3)nn12 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)CN(C2CCSC2)C)C(CO)C1 c1(OCC)noc(C)c1NC(C1C=CCN1C(=O)CC1(OC)CCC1)=O C1(OCCCC)CCCN(N(C)C2CN(C)CC2O)C1 N1(C(C(CCC)O)=O)CCC2(CC1)CN(c1nccc(SC)n1)C2CCO Cc1ccnc(C(=O)NCC2CN(C)CCN2C(=O)C(O)C2CCC2)c1N C(=O)(CC(CC)NC(c1ccnn1CC)=O)NCC(C#C)OC c1(C(C(=O)NC(CC)CNC(=O)CCc2cnco2)C)ccc(OC)cc1C c1(C(=O)NC2(CCCNC(C(C)(C)OCC)=O)CC2)n[nH]c(C)c1Cl CC(CC(N)=O)C(=O)N1CCC(CCN(C)C(c2ncncc2N)=O)CC1 C1(NC(c2onc(CC)n2)=O)CCC2(COC2)N1C(=O)OC(C)(C)C.COC c1(C(C)=O)ccnc(C(N2CC(CO)(NC(C3CCCCN3C(C)C)=O)C2)=O)c1 c1(CC(C(=O)O)NC(CC2CCC(C)C2)=O)cc(F)ncc1Br C(=O)(CCCC(C)C)NCC(c1c(OC)cccc1)NC(=O)CC1CCC(=O)N1 N1(C(c2c(C)nc[nH]2)=O)CCCC(C(C)C(=O)NCCC2CCN(C)CC2)C1 N1(C(C(COC)O)=O)CCc2nc(CNC(=O)C(C)(C)C(C)C)sc2C1 c1(C(=O)NC2CN(C(COCCC#C)=O)C(C)C2)cc(Cl)c2ccccc2c1O N1(c2c(C)c(Cl)ncn2)CC2CC(NC(C3(C(F)F)CCOCC3)=O)CC1C2 c1(C(N(CC(CC)NC(c2cc(C)c(CC)o2)=O)CC)=O)cc(C)n(C)n1 C1(NC(CCSc2n(C)ccn2)=O)CC(NC(c2ccnnc2O)=O)C12CCC2 C1(=CCNC(Cc2cc(C)on2)=O)CCN(C(C2(CC(C)C)CCNC2=O)=O)CC1 Cc1cccc(CC(=O)NCCOCCOCCCNC(C2CC2(F)Cl)=O)c1F CC(C)C(C(=O)NCC(Cc1ccco1)C(=O)N(C)CC1CC1)C(C)C C1(C(C)(C)NC(C(C)NS(C)(=O)=O)=O)CCN(C(c2cncn2C)=O)CC1.C1(C)CC1 C(=O)(C1=C(Cl)CCCC1)N(C(CNC(c1ccc(C#C)nc1)=O)CC)C N1(C(c2cc(C)no2)=O)CC(NCc2c(C)n[nH]c2C)C2(CC2)C1 C1(CCOC)CCCN(C(c2cn(C)nn2)C(=O)NC2CCOC(C)C2)C1 c1(C(=O)NC(C2CCN(C(COC3CN(C(C)=O)C3)=O)C2)C)cc(C)nn1C c1(NC2C(C(C)C)CCC2)nc2ccccc2nc1NCCCc1ccn(C)c1 CC(C(=O)NCc1ccc(C(NC[Si](C)(C)C)=O)o1)C(C)(C)C C(CC(C(=O)NCCOCCN=[N+]=[N-])NC(=O)C(C)CC1CCC1)SC C1(C(N(C(C(=O)NC(CN(CC)CC)C)C)CC)=O)C2CCC(C2)C1C c1(OC)ccc(C(N2CC3CC(NC(=O)C(C)C4CCC4)C2C3)=O)cc1O CN1CCCC(C)(C(N(C2CCCCN(C(c3cccc(Cl)c3F)=O)C2)C)=O)C1 O=S(=O)(c1ccc(Cl)cn1)N1CC2CN(Cc3ccc(CO)o3)C2C1 C1(C(=O)NCC2CCC(NC(CCC(=C)C)=O)C2)CN2CCN1CC2C C(=O)(C(CC(C)C)CC(C)C)NC(C(C)NC(C(CC(C)C)N(C)C)=O)CO CC1(O)CCCCN(C(C2C(C(=O)Nc3ccc(Br)c(Cl)c3F)C2)=O)C1 c1(C(=O)NCC2(C)CCN(C(c3c(CC)[nH]cc3)=O)CC2)cc(F)c(F)cc1N Cc1nc2ccc(C(=O)NC3CCN(C(C4(CC5CCC5)CC4)=O)C3)cc2n1C Cc1c(C(N2CCCOC(CNC(=O)CC3CCCC3O)C2)=O)sc2cncn12 Cc1ccncc1C(=O)N(C1CCCN(C(=O)Cc2ccoc2)C1)C c1(OC)ccccc1C1(C(=O)NCC(C)N(C)C(C2CCC(C)(C)C2)=O)CC1 C(=O)(C(O)CC(C)(C)C)NCC(CC)NC(c1nc(CC)oc1C)=O N1(C(c2c(CC)noc2)=O)CCN(C(c2[nH]cc(C)c2C)=O)C(CC(F)F)C1 C(C(C)(CC)CC)(c1cccc(OCC)c1)NCC1CCCC(C(F)(F)F)O1 c1(C(N2C(CC=C)(C(=O)OC)CCC2)=O)c(F)cc(OC)cc1F c1(C(=O)NCCCCC2CN(C(C(C=C=C)C)=O)C2)ccc(Cl)c(OC)c1F C1(C(=O)NCC(C)N(C(C(c2cccs2)SC)=O)C)CCN(C)CC1.C(C)(=O)NC C12(NC(CC=C)=O)CN(C(c3cccnc3)=O)C(COC)(C1)C2 Cn1nc([N+](=O)[O-])cc1C(N1CC2(CC(NC(=O)C(CO)C(F)(F)F)CO2)C1)=O C1(C(N(C)CC2CCN(C(=O)Cc3nccn3C)C2)=O)Cc2c[nH]cc2S1(=O)=O N1(C(CC2CC(OC)C2)=O)CCSCC1C(=O)NC1CC1(C)C c1(C(=O)NCC(CC=C)NC(=O)C2=C(C)CCOC2)cc(C#N)ccc1F C(C(C(=O)NCCC1CCOC1)NC(c1csnc1C)=O)SCC c1(C(N2C(C3(NC(C4CCCSC4)=O)CC3)CCC2)=O)nc[nH]c2ncnc1-2 N1(C(C(C2CCC(=O)N2)C)=O)CC2(C1)CN(C(=O)C(c1nc(O)n[nH]1)C)C2 C(C1=CCCN(C(=O)CCC2CCCC2)C1)NC(=O)Cc1ccc(OCF)cc1 C12(CCC(C)(C)CC1)CNC(=O)N2.C1(C(C)C)CCCC1C(F)F O=C1NCC(C(N2CC(NC(C34CC(C3)NC4)=O)C2)=O)N1 C(CC(=O)N1CCC(NC(c2cccc(N)c2O)=O)CC1C)(C(F)(F)F)OC c1(C)cc(C(C(CCNC2CN(C(N)=O)C2)=O)=O)co1.N(CCO)C(C)C C(=O)(C1=CNC2=NCCCC2=C1)NCCOC1CN(C(c2c(CC)nns2)=O)C1 C(C(C)(C)CC(F)F)C(N1C(CC#C)(NC(C2C3CC4C(C3)C24)=O)CCC1)=O c1(C(N2C(C(N3CCC(CO)CC3)=O)CSCC2)=O)cccc(F)c1Br C1(C(=O)NCCn2nccn2)CCN(C(c2ccc(Cl)cc2Cl)=O)CC1O C(c1ccc2c(c1)OC(F)(F)O2)=CC(=O)OCC(c1c(Cl)ccc(Br)c1Cl)=O c1(C(=O)NCC(C(C)C)NC(CC(c2ccc(C)cc2)C)=O)cc(Cl)ccc1F C1(C(=O)NCc2cscn2)CCN(CC(C2CCC2)OC)CC1 c1(NC(C2CCCN(C(c3ccnc(C)n3)=O)C2)=O)cc(F)c(F)cc1[N+](=O)[O-] C1(C(=O)NCCCCNC(c2ccc(C#N)o2)=O)CCC(N=[N+]=[N-])CC1 c1(C2C(C(N3CCC(SCOC)C3)C(=O)NC)C2)ccccc1C CN1CCC2(CCN2C(=O)CCCCCN(C(=O)C(F)C(C)(F)F)C)C1 CN1CCC(CC(=O)NC2(CC(=O)N(C3CC4CC4C3)C)CCC2)CC1 C12(NC(C3(C(CC)=O)CC3)=O)CCCN(C(c3ncnn3C)=O)CC1C2 Cc1c(Br)sc(CNC(c2cc3n(n2)CCC3)c2nnnn2CCC2CC2)c1C C1(CNC(CN(C2CCSC2)C)=O)COCCN1C(=O)Cc1cncc(F)c1 C12(C(N3CC(CC)OCCC3)=O)CCCC1CN(C(C1CCCC(CF)C1)=O)C2 c1(C(N2CC(O)(C(C)NC(C3CCC3(F)F)=O)C2)=O)cccc(C(F)F)c1F C(CC)(CCC(=O)NCC(O)C(F)(F)F)NC(C(C)OCCCC)=O c1(NC(CC#C)(C)C)cc(Br)ccc1C(=O)OC N1(CC)N=C(C(=O)NC2CCN(C(=O)C(c3cccnc3)O)CC2F)CCC1=O c1(CC(=O)N(C(C)CCNC(C2CC(F)C2)=O)C)ccnc(O)c1 C(CCCNC(c1cccs1)=O)(c1ccccc1)NC(CC1(CC)CCC1)=O N1(C(C2C(C(C)(F)F)C2)=O)CCC2CCCC12CNC(c1coc(Br)n1)=O C1(C#N)(C(N2CC(COC)(CNC(=O)C(=O)NC3CCC3(C)C)C2)=O)CC(C)C1 c1(CC(=O)O)cc(C(F)(F)F)nn1C.CCCCN(CC)CCNC(=O)CO Cc1oc(C#N)cc1C(=O)NC(C1CCCCC1)C(=O)NC1(C)CS(=O)(=O)C1 c1(C(=O)NCC(CNC(CC2(C)OCCO2)=O)(C)O)ccc(OCC(F)F)cc1 C1(C)(C)C=CCCC1.n1(CC)nnnc1C(c1noc(C2CC2)n1)NCC1CC1 CC1(C(=O)NC2CCC(NC(=O)C(O)Cc3cnc[nH]3)CC2)CCCCO1 c1(C(=O)NC2CN(C(C(C)Cc3ccccc3F)=O)C2)cc2cccnc2o1 C(=O)(C1=CCCOCC1)NC1CCN(C(c2n(CC#N)ncc2)=O)CC1O CCCCCC(=O)N(C1CCN(C(=O)CC2OCCC2C)CC1)C C1(C(N(C)CC2(Br)CC2)=O)CCCCC1CNC(=O)CN1CCSCC1 C1(C(N2CC(C)C(CNC(=O)CC3CC3)CC2)=O)CC2C=CC1C21CC1 C1(C(=O)NCc2nc(-c3cn(CC4(CO)CC4)nn3)sc2F)CCC(C2CC2)C1 C1(CC(=O)NCC(CCC)NC(=O)C(C)(C)O)CCCC(F)(F)C1 C(c1cccc(N)c1)=CC(=O)N(CCNC(=O)CCC1CCN(C)CC1)CC C12(C(N3CCC(NCC(C)NC(C(c4cnccn4)C)=O)C3)=O)CC(C1)C(C)O2 CC1(C)CC(C(=O)NCCOCCC(=O)NCC2CC3CCCC3C2)CCO1 c1(C(N2C3CCC2C(C(=O)NCCN2CCCC2)C3)=O)ncc(Cl)cc1F c1(C(=O)NCC(CCNC(C(CC(=C)C)C)=O)O)cc(C)nc2cc(Cl)ccc12 CN1Cc2c(C(=O)NCc3nnc4n3CCOC4)cccc2NS1(=O)=O N1(C(C(CNC(c2cc(C(N)=O)c[nH]2)=O)N(C)C)=O)CC2(CCOCC2)C1 N1(C(c2nc(COC)oc2)=O)CC2CCN(C(=O)C=C3CCCCC3(C)C)C2C1 c1(N(C)CCc2ccc[nH]2)c(Br)cc(C(F)(F)F)cc1I.C12CN(C1)CC2O O=C(CCC(=O)N1CCNOCC1)SC1CCCCCC1 CC1(C)CC=C(C(=O)N2C3CCC2C(F)C(NC(=O)CC2CC2(C)C)C3)CC1 C(=O)(CC(C)C(F)(F)F)N1CCCC(C)(NC(Cc2ccc(SC)cc2)=O)C1 c1(C(=O)NC(C(C(C)C)NC(C2C(C)(C)C2(C)C)=O)C)noc2ncccc12 N1(C(=O)OC(C)(C)C)CC2CC(C(N3CCCC(C(C)(F)F)C3)=O)CC(C1)C2=O c1(C(=O)NCCC(C)(C)NC(C2CC=C(C)CC2)=O)cc2n(n1)C(C)CCC2 C1(NC(C2(CCOC)CCC2)=O)CN(CC)CCC1O.C12(CCC1)C(=O)N2 C1(NC(=O)NCC(CCSC)N)CCC(C)(C)CC1Cc1ccccc1.SC N#CC1CCN(C(C2CC(Nc3cc(C(=O)Nc4ccccc4)ncn3)C2)=O)C1 c1(C(N2CCCC(N(C(=O)Cn3ccnn3)C)C2)=O)scc2c1CCCC2 C1(NC(C2CCC(C(C)C)CC2)=O)CCCCN(C(C2(F)CCOCC2)=O)C1 C1(C)(CCNC(c2c(C)onc2)=O)CCN(C(C2CCC(C(C)(C)O)CC2)=O)C1 N1(CCOC)CCCCC1CNC(=O)C(=O)NC1CCN(C(C)C)C1 c1(NC(C2N(Cc3ccc(C)c(Cl)c3)CC(C)C2)=O)cccc([N+](=O)[O-])c1Br C1(CNC(c2c(C(C)C)ncs2)=O)(CO)CCN(C(c2cc(C3CC3)ns2)=O)C1 C=CCC(CC=C)C(=O)NCC(C(C)C)NC(c1cnn(CCO)c1N)=O N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CC1CN2C(=O)CC(=O)c1ccco1 CC1(C)CCCC(CC(=O)OC2CCC(CS(C)(=O)=O)CC2)O1 c1(C2C(C(=O)NC3(CC(=O)NC4CN(C)C4)CCC3)C2)ccc(Cl)c(C#N)c1 CC1CCCN(C(c2ns[nH]c2=O)=O)C1CCNC(c1ccc(N)c(F)n1)=O c1(OC)c[nH]c(C(C(=O)NCCN2CCC(CO)CC2)N(C)CC2CC2)cc1=O N1(C(c2cccc(-c3cn(C4C(OC)COC4)nn3)c2)=O)CCOC2(CCC2)C1 C(=O)(C(O)CCC(C)C)N1CCC(N(C(c2nc(OC)c(F)cn2)=O)CCO)C1 CCCC(CC)CCC(=O)N1CCC(N(C2(C3CCCO3)CC2)C2CC2)CC1 n1(CC(C)(F)F)ccc(NC(N2CCC(Br)C2)=O)n1 c1(C(=O)OCC)cc(C)c(O)nn1.C1(=O)CCC(=O)CN2CCN1CC2C C(N(O)C(=O)Cc1cccc(Cl)c1)c1cn(C(C)(C)C)nn1 N1(C(C2N(C(C3N(C)C(=O)CCC3)=O)CC(O)C2)=O)CC2C=CCC(C2)C1 CC1CC(Nc2nc(C3CC3(F)F)cs2)CCN1 C1(OCC)CCCC(NCc2nc(-c3cnccn3)no2)C1 CC12CCC(C(=O)NC(CNC(=O)C(F)=CC3CC3)CO)(CC1)CO2 N1(C(CCOCCOCCOC)=O)CC(NC(=O)C(F)(F)CO)C(C)(C)C1 C1(C2CC2)(NC(CCCCC=C)=O)CCN(C(c2noc3c2CCCC3)=O)C1 CC1(C)CCC(CNC(c2cc(F)c[nH]2)=O)(NC(C2CCC3(CCC3)O2)=O)C1 Cc1ccnn1C(C)C(=O)NC(C1(O)COC1)C c1(COC)ccc(C(N2CCCC2C(=O)NC2(C(C)C)CC2)=O)cc1 C1(CNC(C(F)=CC)=O)CCCC2(CN(C(=O)C(C(C)(C)C)N(C)C)C2)O1 C(=O)(CC(F)(F)F)N(CC)CO.N1(C(C(C)OC)=O)CCN(C(=O)CC2OCCCO2)CC1 c1(C(=O)Nc2ccnc(-c3cnn(CC4CC4)c3)c2)onc2ccccc12 C1(c2c(OC)cccc2)CN(C(=O)C(F)F)CCN1C(=O)CCCC(=O)N(C)C CC1(C)CC(CC(=O)NCc2cccc(CNC(=O)CSC(F)F)c2)NC1=O C1(CNC(C(CN(C)C)NC(CCN(CC)CC)=O)=O)COCC1(C)C N1(C(CC(C)N(C(C(=O)NC(C)=O)=O)C)=O)CCC(N(C)C)CC1 C1(NC(c2ccc(CO)o2)=O)CCCN(C(C2CC(n3ccnn3)C2)=O)CC1 c1(C(N(C2CN(C(Cc3cc(C)[nH]n3)=O)CC2F)C)=O)cc2nccn2c(O)n1 C(=O)(CCCc1sccc1C)NC(CC)CNC(C1(COC)CCCC1)=O C12(C(=O)NC(C)CCCNC(=O)CC3CCC(C)CC3)CCCC1CC(=O)CC2 C(=O)(C1=NOC(C)C1C)NCCCC1OCCN(C(C(COC)(C)C)=O)C1 CC(C)S(=O)(=O)C(C)C(=O)N1CCC2(C1)CN(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 Cc1cccc(C)c1NC(=O)NC1CC1NC(=O)C(C)NC=O CCC(C(=O)NC(CNC(c1ocnc1C1CC1)=O)C1CCC1)N(C)C C(CCCC(=O)NCc1occc1C(N1CCOC(C(C)C)C1)=O)OCC C1(NC(C(n2c(C)cc(C)n2)C)=O)CC2CC1CN(C(c1cccnc1O)=O)C2 C1(C(=O)NCC2(O)CCN(C(=O)CNS(=O)(=O)C3CC3)C2)C2CCCCCC12 c1(-c2ccc(C)o2)nc(C)c(C(=O)NC2(C)CN(C(C3CC3F)=O)C2)s1 c1(NC2(C)C(C)C2)ccc(C(=O)N(CCCN2CCOCC2)C)cc1 c1(CC)nc(C)oc1C(=O)NC12CC(C1)N(C(C1CCOC1C1CC1)=O)C2 C(=O)(CCC(F)(F)F)N1CCC(C(C(=O)NC2C(CC)CCC2)C)CC1 C(=O)(CCCC(CC)NC(=O)Cc1c(C)cnn1C)NCCCC=C C1(O)(CCNC(=O)COC2CC=CC2)CCN(C(C2CC3CCC3C2)=O)C1 C1(C(N(C2CCN(C(=O)CCc3cnccn3)CC2)C)=O)CC(=O)N(C2CC2)C1 c1(C(=O)NCC2CC(NC(C3C(c4n(C)nnc4)C3)=O)C2)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC2C3CN(C(C(=O)NC)=O)CC2C3)cnc2n(c1=O)CCS(=O)(=O)C2 c1(C(N2C(CN(C(c3ccc(C=C)cc3)=O)C)CCC2)=O)cncc2[nH]ccc12 C=CCCCC(C(=O)NCC(C)C(F)(F)F)NC(C1COCOC1)=O c1(CNC2CCC(C(=O)Nc3cccc(C#C)n3)OC2)n[nH]c2ccc(Br)cc12 c1(C(N2C(C(=O)NC(C=C)CO)C=CC2)=O)ccc(F)c(Br)c1 c1(CCCC(=O)OCc2ccncc2Br)c[nH]c2ncccc12 c1(C(C)NCC(=O)NC(c2ccccc2)=O)cccc(Cl)c1 C(c1ccc(OC)c(F)c1)=CC(=O)NC(C(=O)OC)Cc1cn(CC(C)C)nn1 CC1=C(C(=O)N2CCCOC(CNC(C3(F)CCC3)=O)C2)CCO1 N(C1CCc2ccc(Cl)cc21)C(CC)C(=O)OC(C)(C)C N1(C(Cc2nc(C)sc2)=O)Cc2ccccc2C1CNC(=O)CCC(C)(C)F c1(CC)c(C(=O)NCCCNC(=O)COc2ccc(OC)cc2)cnn1CSC C(C)(C(=O)NCCCCO)N(CCC)C(C1CCO1)=O C1(NC(C(CSC)c2ccccc2)=O)CCCCC1NC(=O)C=Cc1cncn1C C1(NC(Cn2ncc(CC)c2)=O)CCC(C)(C)CC1CNC(=O)C=C1CCC1 C(=O)(C1CCCCc2ccccc21)N1CC(NC(=O)CCN2CCCC2)C1 C12(NC(C(C)NC=O)=O)CCC(C1)N(C(=O)Cn1[nH]cnc1=N)C2 CC(=O)C(C)CC(C)C(=O)N1CC(C(=O)N(C)Cc2cccnc2)CC(C)C1 C1(CNC(C(CCOC)C)=O)CCCCN(C(c2cc(C3CCC3)no2)=O)C1 c1(OC)ccc(C(=O)N(CCN(C(=O)C(C(C)O)N(C)C)C)C2CC2)c2ccoc12 c1(C(N(C(C2CCCCC2)CNc2ncc[nH]2)CCC)=O)nc(C(C)C)oc1C C(N=c1ccc2nnnn2[nH]1)C12C(CN(C(C3=CC(C)(CC)C3)=O)C1)CCCC2 C(CCCCCN(C)C(C1CCOC(C(C)C)C1)=O)NC(C(CC)NC(C)=O)=O Cc1nc(CC(=O)N(CC(C)O)CCNC(c2cccs2)=O)cs1 C1(C(C)NC(=O)OCC(C)(C)C)CCCN1CCC1OCCO1 C1(NC(=O)COCC2CCC2)CCCC2CN(C(c3nccc(Cl)c3F)=O)CC12 N1(C(c2c(CC)c[nH]c2)=O)CCN(C(=O)CC2=CCN(C)CC2)C(C)CC1C CC1(C)CC(NC(c2cccc(Cl)c2F)=O)CN1C(C1CCC(=O)C1)=O CCS(=O)(=O)CC(=O)NCC(CC)CC(=O)NC(CO)CCCO c1(CC(=O)NCC2(NC(c3n[nH]c(C)c3Cl)=O)CCOCC2)ccnc(F)c1F C(C)(C(CC(=O)N1CC=CC1CF)NC(c1cnc(C)cc1C)=O)OC CC1CN(C(c2ccnc(N(C)C)c2)=O)CCC1C(=O)N(C)CCN(C)C C(C(=O)N1CC(O)CO1)n1cc(NC(CNS(C)(=O)=O)=O)nn1 N1(C(C2CC(CNC(C(C)OC)=O)OC2)=O)CCCN(C)CC1 c1(C(N2CC(CC(C)NC(c3c[nH]c4cccnc34)=O)C2)=O)ccc2[nH]ccc2n1 Cc1n[nH]c(=NCC(C)(C(C)C)NC(=O)CC2CCNC2=O)s1 c1(-c2onc(C)n2)ccc(C(=O)NC(C)CN(C)C(c2nocc2Cl)=O)cc1 C(CC(C)(C)CC(=O)NC1CCN(C(=O)CC2CCOC(C)(C)C2)C(C)C1)OC C1(NC(c2ccn(C)c2)=O)COCCN(C(c2cc(C(C3CCC3)=O)c[nH]2)=O)C1 CC1CC(NC(C2CN(C(=O)CCS(C)(=O)=O)CC2C)=O)CC(C)(C)C1 CC1=NN(C)C(=O)C1CC(N1CCCCC1CNC(c1nc[nH]c1C(C)C)=O)=O C(=O)(CCCCC(=O)NC)N1CC2CC(NC(C=CCC)=O)C2C1 C12(C(=O)NC3CC(C)N(C(=O)C(=O)Nc4ccccc4O)C3)CC3CC1C2C3O CC1=NOC(C)(C(N2CCC(C(C)(C)CNC(c3cc(C)cnn3)=O)CC2)=O)C1 c1(C(N2CC2=O)=O)cnc2c(Br)n[nH]c2c1.c1(C(C)(C)C)cnc(C2CCC2)o1 C(=O)(C(O)CC(C)C)N1C(C(=O)NC2(COC)CCC2)C2CC2C1 C(=O)(CCCC(=O)NC1CC1)NC(C(=O)NCC1(O)C(C)CCC1)CO c1(OC(c2cn(CCOc3ccccn3)nn2)=O)ccc(F)c(Cl)c1 Cc1cc(C(=O)NCC(C)CNC(=O)CC2CSCCS2)cc(N)c1Cl c1(OC)cnc(F)c(C(=O)NCC(n2cc(-c3cnccc3Cl)nn2)C)c1 C1(C(=O)NC(CC(=O)OC)C)CCN(C(=O)CCc2nccs2)C(C(C)C)C1 C1(C(=O)NC(C(=O)NCCc2c(C)n[nH]c2)(C)C)CCCN(C)C1 C1(CC)C(NC(c2cccnc2C)=O)CCCN1C(=O)CN1CCC(OC)C1 C1(C(=O)NCC(C(C)C)C)CC2CC2N1C(c1csc(Cl)c1)=O c1(N2CC(CNC(C(C)(C)CC)=O)OCCC2)nc(C(=O)NC)nc2c(C)csc12 C1(N(C(c2c(C(C)C)cccc2)=O)C)CC2CCC(C1)N2C(C1(N=[N+]=[N-])CC1)=O N1(C(C(C)CCO)=O)CCN(C(=O)Cc2csc(NC=O)n2)CC(O)C1 CCC(C)CCCCC(=O)N1CCC(NC(=O)CSc2ccccn2)C(C)C1 Cc1cn2c(C(N3CC(CCCC)CC3C(=O)O)=O)c(Cl)nc2s1 C(=O)(C(C)CCO)NCC(C(C)C)NC(=O)C(c1ccc(Cl)s1)C c1(C(N2CC3C(NC(C(C)(C)SC)=O)C3C2)=O)cccc(C(C)C)c1O C1(CC(=O)NC(CN(C(c2ccoc2CC(N)=O)=O)CC)C)CCCS(=O)(=O)C1 C1(CCNC(C2CC(OC(F)F)C2)=O)CCN(C(=O)CSC2CCCCO2)C1.OC C1(C(=O)NC(C2CCCN(C(C=CSC)=O)C2)C)CS(=O)(=O)CC(=O)N1 C1(NC(c2ccc(SC)cc2)=O)CN(C(=O)Cc2nonc2C)C2CCCCC12 CC(C)C(C(=O)NCC1(C)CC1)C(C)NC(c1cnn(C)n1)=O N1(C(C2CCN(C(COC3(C#C)COC3)=O)C2CC)=O)CCC(OC)C1(C)C C1(NC(C2(Oc3ccccc3F)CC2)=O)C2CN(Cc3ccccc3)CC12 N1(C(CCSC)=O)CCC(NC(C2CN(C)CC(C)O2)=O)CC1C CC(C(=O)NNc1ccc(Br)nn1)c1c(F)ccc(C)c1F c12ccc(cc1F)Oc1noc-2n1.c1(OC)ccc(C(c2ccccc2)O)cn1 C1(C(CNC(c2ccoc2CC(N)=O)=O)C)CCN(C(C2CC2C(F)F)=O)CC1 C1(NC(c2ccc(CC)cc2)=O)CN(C(c2cccnc2)=O)CCC1(F)F N1(C(C(C)OCCOC)=O)CCC(C)(CNC(=O)CCc2nc(CO)no2)CC1 C1(O)(CC(=O)NC2C(C)(C)C2CO)CCCOC1.C1(=O)CCCn2cc(nn2)CN1 CN1CCN(C(C2OC3CCC2CC3)=O)CC1CNC(=O)CCN1CCC1 c1(C(=O)NC2C3CN(C(CC=C(C)C)=O)C2C3)cc(S(N)(=O)=O)c(Cl)cc1Cl c1(C(N(C2CCN(C(C3CC(C)=NO3)=O)C2)CCC)=O)ccc(COC)cc1 C#Cc1ccc(C2N(C(=O)OC(C)(C)C)CCCC2NC(=O)C(F)F)cc1 C1(C(=O)NCCNC(Cc2cn(CC)nc2)=O)CCCS1(=O)=O N1(c2nnc(-c3c[nH]c(Br)c3)n2CCC2CC2)CCN(CCC2CCCO2)CC1.FC(F)O CCC(CC(F)F)C(=O)N1CC(CNC(c2cnoc2C(C)C)=O)CC1(C)C N1(C(C2CCS2(=O)=O)=O)CC2CCC1CN2c1ccnc(Cl)n1 c1(C(=O)NCCCC(c2cccs2)NC(C(C=C)O)=O)c(F)c(N)cc(F)c1F C1(C(=O)NCC2N(C(C3(F)CC3)=O)CCC2)CC12CCOc1ccccc12 c1(OC)cc2ccc(CC(=O)N=c3cc(C)n(CCO)[nH]3)nc2cc1F c1(C(=O)Nc2ccc(-c3cnn[nH]3)cc2)ccc(O)cc1Cl c1(NC(C(C)N(C)C)=O)cccc(CNC2CCN(C(=O)CCCC3CC3)C2C)c1 c1(C(=O)NC2CCC(NS(CC=C)(=O)=O)CC2)ccc(F)c(OC)c1F c1(C(N2CC(OC)CC(NC(C(C=C)(C)C)=O)C2)=O)ccc2nn[nH]c2c1 N1(C(C(C)OC)C(=O)NC(C)C)Cc2[nH]c3ccccc3c2CC1C CC(C)(C)CS(=O)(=O)N1CCCC(c2nc(C(=O)O)cn2C)C1 C1(C(N2CC(NC(=O)Cc3nnco3)C2)=O)CCCC12OCCO2 N1(CCNC(Cc2cc(C)no2)=O)CCN(C(C2CCCC23CC3)=O)CC1 c1(C(N(CC(CN(C(C)=O)C)O)C)=O)n[nH]c2ccc(Cl)cc12 c1(CC)ccc(C(N2CCC(NC(c3cc(COC)no3)=O)C2(C)C)=O)cc1F N1(C(C2N=C(C)SC2)=O)CCCCC2(C1)CN(C(=O)CCCN1CCCC1)C2 NS(=O)(=O)c1cc(C(=O)OCCC2CS(=O)(=O)C2)c(Cl)c(F)c1 C1(C(=O)OC)C(C(=O)NCC2(NC(C34CCC(C3)C4)=O)CC2)C1(C)C CC(C)(C)CCCC(=O)NCC1CCC(C(N2CCC(CCO)C2)=O)C1 c1(C(N2CC(C(C)NC(c3c(C(C)C)nns3)=O)C2)=O)cc2ccsc2[nH]1 Cc1ccc(C=CC(=O)NCC2(CNC(=O)C(C)O)CCCCC2)cn1 N1(C(c2cnc(C)nc2C)=O)CCCC2(NC(c3cnc(C)[nH]3)=O)CCCC12 Cc1ccc(N)cc1C(N1CCC1C(C1CC1)NC(=O)Cc1ccc(Cl)s1)=O N1(C(=O)OC(C)(C)C)C(C(=O)NC2(Cl)CC3CCC2O3)CCC12CC2 N(C1CCc2c(Cl)cccc21)C(C(N1c2ncc(C(=O)OC)cc2CC1)=O)=O C1(C(N(C)CC2CCN(C(C3CC(C(=O)OC)C3)=O)C2)=O)CCC(C)(C)OC1 c1(NC(CC)CCCO)ccc(S(=O)(=O)N2CCCC(SCC(C)C)C2)cn1 C=CC1(C(=O)NCC(O)C(=O)N(C23CCC(CC2)CC3)C)CCCCC1 c1(NC(C)=O)ccc(C(=O)NC(C)CNC(C2(C#N)CC(C)C2)=O)c(Cl)c1 C1(CN(C(=O)CCC(=O)NC)CC)CCCCN1C(C1CC2CC2C1)=O N1(S(c2ccc(C(=O)OC)nc2)(=O)=O)CCCC2(CCN(C(=O)CSC)C2)C1 c1(NCCCC(N)=O)nc(N2CCSCC2)nc2scnc12 C1(NC(CCOc2ccc(CC)cc2)=O)CC2CCC1N2C(=O)Cc1cnns1 C(=O)(CCCS(C)(=O)=O)NC(C1N(C(CC(CC)C2CC2)=O)CCC1)(C)C CC(C)C(C(=O)NC1CN(C(=O)C(C)C2CC2)CC1C)NC(c1cccs1)=O N1(CCCNC(C2C(OC(C)(C)C)C2)=O)CCN(C(c2ccc(F)s2)=O)CC1 CCC(C)(C(=O)NC(C)C(=O)NCCC(C)N1CCC1)OC N1(C(c2c(C)n(C)cn2)=O)CC2CN(C(=O)Cc3ccc(F)cn3)CC2(C)C1 c1(C(=O)NCC)c[nH]nc1C(F)F.C1(CCCSCC(=O)N)CC(O)C1 c1(OC)cc(Cl)c(C)cc1COC(=O)C(F)(F)CC(C)C c1(CN2CCCC(C(F)(F)F)(OC)C2)c[nH]c2cc(-c3nn[nH]n3)ccc12 CC1CN(C(=O)CC(F)(F)F)CCN1C(c1cc(Cl)c(Cl)[nH]1)=O N1(C(c2cc(C#N)oc2)=O)CCCC2(CCCN2C(c2ccc(Cl)nc2O)=O)C1 N1(C(c2[nH]cc(OC)c(=O)c2)=O)CCCC2CN(c3cc(O)nc(O)n3)CCC12 Cc1cnc2n1CC(C(=O)NC(C)CN(C)C(c1cc(F)c(F)cc1N)=O)CC2 CCCC(C)(C)C(=O)NCCC(C)NC(C1CCC12CCOCC2)=O CCCC(CCC)CCCC(=O)N1CC(CCNC(=O)CN(C2CCSC2)C)C1 C1(C(=O)OC)CC(=O)CN1C(c1c(O)noc1C)=O c1(CCC(=O)NCC(CNC(C2=C(C)OCC2)=O)C)cccc(S(N)(=O)=O)c1 O=C(C(Cl)=CCl)NC1CCC(CCNC(C2CCC(C(F)(F)F)O2)=O)C1 CCC(CSc1ccc(F)cc1)CC(=O)N1CCC1CNC(C1(CSC)CC1)=O CN1CCc2c(NC(=O)NC3(c4ccncc4)CCC3)cccc2C1=O Cc1ncc(CC(=O)NCC2(O)CN(C(C3CC3[N+](=O)[O-])=O)C2)[nH]1 C1(CCC(=O)NCC(C2CCCC2)N(C(C2(SC)CC2)=O)C)CCC(=O)N1 C(=O)(C1=CCCOC1)NC(CCNC(C(C(C)C)N(C)C)=O)C c1(N2CCCC(CN(C(=O)C=Cc3cocn3)C)CC2)c(Br)cccc1[N+](=O)[O-] c1(NCc2cc(C)ns2)cc(NCC(Cl)=CCl)ncn1 c1(C2C(C(N3CC(C)C(n4cc(C5CCC5)nn4)C3)=O)C2)ccc(F)cc1Cl CC(C)CCN=C(NCc1ccc(Br)o1)NC(C1CCCO1)C C(=O)(C(C)(C)CC(=O)NC(C)CNC(c1ccccc1C(C)(C)C)=O)OCC CCC(C)CCCCC(=O)N1CCC(C(F)(F)F)C(NC(=O)C=C(C)C(F)F)C1 C(=O)(C(C(C)C)C(C)C)N1CC(C(=O)Nc2cnc(SC)s2)C(n2cccn2)C1 c1(CC)cc(C(=O)NCC2CCC(C(=O)NCCC(C)(C)F)O2)n[nH]1 O(C=C(C#N)C(=O)N1CC(NC(c2cc(C3(C)CC3)on2)=O)C(C)(C)C1)CC C1(Nc2c(C)cnn2CO)COc2ccccc2C1C c1(CC(=O)N(CCCCNC(=O)CSC)C)ccc(C2CC2)cc1.CO N1(C(=O)NC2(O)CCC(CC)C2)c2ccc(Br)cc2NS1(=O)=O C(C(COC)C(=O)N(CCNC(C1CC2CCC1C2)=O)C(C)C)OC c1(CC)ccc(C(=O)NCCCOCCNC(C2CC2(F)F)=O)c(Cl)c1OC C1(CC2C(CC)CCCC2)CC(O)C12CCC2.C1=CC(=O)NC(=O)CC1 c1(C(=O)NC2C(NC(COCCCC(C)C)=O)CCOC2)cn2c(n1)CCC2 C(C)(C(=O)N(CCCNC(=O)CNC(=O)Cn1cncn1)C)=CC Cc1ccc(C(=O)NCC2CN(C(c3cnnn3C(C)C)=O)CCO2)c(C)n1 C#Cc1ccc(C(N2CCC3CC23C(=O)NC(CSc2nc[nH]n2)CC)=O)cc1 N1(C(c2c(C(C)(C)C)ocn2)=O)CC2C3CCC(C(NC(=O)CCCF)C3)C2C1 N#CCCCC(=O)N1CCCC1CC(N1CC(N(C)C2CC2)C1)=O CC1CC(NC(=O)CCNC(c2cnn(C)c2)=O)CN(C(C2CCCCC2)=O)C1 C1(C)(C(=O)NCCC(CC)(C)NC(C2COCCO2)=O)CCCN(C)C1 C1(N(C(c2cc(CC(C)C)[nH]n2)=O)CC)CCCN(C(=O)CN=S(C)(C)=O)CC1 C1(NC(COCCOC)=O)CCC12CCN(C(=O)C(C)Cn1ccnc1)CC2 c1(NCC2(OCC)CCOC2)nc(N(CC(C)N(C)C)C)c2c(n1)c(C)nn2C c1(OCC)cccc(C(=O)N(C)CCN(C)C(C2CC(C)OC2=O)=O)c1 CCC(CC(F)F)C(=O)NCC1(NC(c2ccn(CC)c2C)=O)CCOCC1 C1(CNC(C(=O)NCC)=O)C(C)CCN1C(c1ccc(SC)o1)=O C1(C(N2C(CNC(COCCCCC)=O)CC2)=O)CCCC(F)(F)C1 C1(NC(CN(C2CCSC2)C)=O)CC(C2CCN(C(C3CC3F)=O)C2)C1 CC1C(C)N(C(c2cccc(C#N)c2)=O)CCN1C(=O)Cc1cccs1 c1(C(C(=O)NCC(C)C)N(CCCOC)CC2CC2)nc(Br)ccc1OC n1(CC)cc(Br)cc1-c1nc(C2CC=CCC2)nn1CC1CCS(=O)(=O)C1 C1(CNC(C(C)Cc2cnn(C)c2)=O)CN(C(c2cncc(F)n2)=O)CCCO1 C1(CNC(N(C)CC2CC2C)=O)C=CCC1 O=S1(=O)c2ccc(cc2Br)N1.c1(CNCc2ncccn2)ccc(F)cc1F C(=O)(C(O)CCC(C)C)NC1C(OC)CN(C(=O)COOCc2ccccc2)C1.O C1(NC(c2cc(CO)on2)=O)CCN(C(=O)CSC(F)F)CC1F Cn1cc(C(C2CCC(C)C2)=O)c(NCCO)n1.C(=O)(N)NCCO.C1CO1.O.C c1(CCC(N2CC(NC(c3c(C)[nH]cc3)=O)C(C)(C)C2)=O)cccc([N+](=O)[O-])c1 CCCCC(C)(C1CCCO1)NC(=O)CSCc1nnc(C)o1 C1(CC(=O)NC(C2CCN(C(C3CCC3(C)C)=O)CC2)C)CCC(=O)NC1 Cc1n[nH]c(=NC2C3C4CCC4C3C2)o1 C1(NC(C2CC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)CCNC(=O)CC1 c1(C(=O)NC(CC=C)CNC(c2nnn(C(C)(C)C)n2)=O)cccc2[nH]ccc12 c1(C(N2CC(C(=O)NC(CC)CSC)C(C)(C)C2)=O)ccc2cncn2c1 c1(C(=O)NCC2CC(F)CN2C(c2cc(Br)n[nH]2)=O)csc2ccncc12 C1(C(=O)NCCC(C)(C)NC(c2cc(C(C)(C)C)ccn2)=O)CCC2C1C2(F)F C1(C(C)S)CCN(C(=O)C=CC(N2CCOCC2)=O)CC1.C1(C)CCCCO1 C1(OC)C(NC(C2CCN(C(=O)C(=O)NC(C)C)CC2)=O)CC12CCC2 N1(C(CCCOC(C)(C)C)=O)CC2(CCCCN(C(C3(Cl)CC3(F)F)=O)C2)C1 CC(C)(C(=O)N1CCC(NC(c2cnn(C(C)(C)C)c2)=O)C(CO)C1)S(C)(=O)=O C1(NC(C(CCSC)O)=O)CCC2CCN(C(C3CC34CCSCC4)=O)C1C2 C1(C(=O)OC)CN(C(=O)NCc2cnc(Br)c(OC)n2)CCS1(=O)=O CC1(C)CC(=O)NC1CNC(C1CCC(CNC(=O)C(C)(Cl)Cl)O1)=O CC1CCCC=C1C(=O)NC1C=CCN(C(c2ccc(F)o2)=O)C1 C1(c2ncc(C)s2)CCCCN1C(c1cccc(Cl)c1)C#N C1(NC(C(=O)NCC2(N(C)C)CC2(C)C)=O)Cc2ccccc2NC1=O C1(C(F)F)(CNc2nc(C3CCCO3)n[nH]2)CCNC1 N1(C(COCCC=C)=O)CCCC(CCC)(NC(c2cccn2C)=O)C1 n1(CC(=C)C)c(N2CCC(c3n[nH]c(C)n3)CC2)nnc1C1CCCCO1 C1(NC(c2ccncc2)C(=O)OC(C)C)CCCN(Cc2cccc(F)c2)C1 Cc1sc(C)c(C(=O)NCC2(NC(c3cnc(C4CC4)[nH]3)=O)CCOC2)c1C#N C(=O)(C(F)(F)c1cscc1Br)N(C(C)CNC(=O)CC1(C)CCC1)C C=CC(F)(F)C(=O)NCCCC(C)NC(C1CN(C(C)=O)C1)=O Cn1cncc1C(=O)NC1CN(C(C2C(c3ccccc3)C2(C)C)=O)C1 N1(C(CCC=CCC=C)=O)CC(OC(F)(F)F)C(COC)C1.C1(=O)C(C)ON1 Cc1ccc(CN2CC3CC3(C(=O)NCC3CC3C3CC3)C2)cc1Cl c1(OC)ccc(Cl)cc1S(=O)(=O)N1CC2CCN(C(=O)OC(C)(C)C)C2C1 C(CN=c1cc(C)c(S(=O)(=O)N2CCN(C)C(C(F)(F)F)C2)c[nH]1)N(C(C)=O)C C1(C)CN2CCC1CC2.C(CCOC)(C(=O)NCCOC)NC(CN(C)CC)=O c1(CCC(=O)NCC(CO)NC(C(CC)C2CCOCC2)=O)cccc(C)c1 c1(CN(C(=O)C(N2CCCC2c2ccsc2)=O)C)ccc2c(c1)n(C)c(=O)n2C c1(NC(N2C(C)(CNC(=O)OC(C)(C)C)CC2)=O)ccc(-c2nncn2C)cc1 N1(C(c2c(C)nc(COC)s2)=O)CCN(C(=O)CC(C)SC)CC1CO C1C2CC(C(CCC)CC(=O)N(CCN(C)C)CCO1)C(=O)N2 N1(C(c2conc2C2CC2)=O)CCN(C(C2CCC2n2ccnc2)=O)CC1CF C1(C)(C(N2CC(n3cc(CN(C(=O)CC4CC4(C)C)C)nn3)C2)=O)COCCO1 N1(C(C2(C=C)CCN(C(=O)Cn3cccc3)C2)=O)CCCC(C)(C)CC1 C(C(N=c1[nH]nc(C(F)F)s1)c1ccc(NC(=O)C(F)(F)F)cc1)(OC)OC c1(C(=O)NCC(CCCC)NC(=O)C(C(C)C)NC=O)nc(C)c(C)nc1C C1(CC)C(C(=O)NCCN2CC(C)(O)C2)CCN1C(=O)C=C1CCCCC1 CC1CCC(NC(=O)CC2CN3CCC2CC3)CN1C(c1ccccc1)=O Cc1c(NCC(C)(C)C)ncnc1NC1CCC1n1ccnc1 C#CCCC(O)C(=O)NC1(CNC(c2sccc2CN(C)C)=O)CCOCC1 c1(C(C2COCCO2)NC(=O)NC(c2onc(C)n2)C)ccc(F)cc1 c1(C(=O)NC(C(=O)Nc2cccc(OCC)c2)(C)C)ncc(Cl)cc1Cl C#Cc1ccc(-c2nc(-c3ccc(Cl)cc3)nn2C)nc1 N1(C(COCC)=O)CC(CNC(c2csc(C(C)=O)n2)=O)OC(C)(C)C1 c1(OC)nccc(-c2cn(CC34CC3CN(C(=O)C(C)CC(N)=O)C4)nn2)c1F c1(CNC(CSC(C)C)=O)ccc(C(=O)NCC2(O)CCN(C)C2)cc1 C1(C(=O)NC2CSC(C)C2)(SC)CN(C(C2CS(=O)(=O)C2)=O)C1 C1(CNC(c2c(OC)nsc2)=O)N(C(C2CC2F)=O)CCCC1(C)C C=CCC(CC(C)C)C(=O)N1CCC(CNC(=O)C=CCN(C)C)C12CC2 c1(CNC(c2n(C)ccc2)=O)nc(CNC(C2C(C3CC3)C2(F)F)=O)cc(O)n1 Cc1cc(C)c(CC(=O)NCC2CC(CS(C)(=N)=O)C2)c(C)c1Br N1(C(C(C(CC)O)C)=O)CC2(CCCCN2C(c2nc(Cl)sc2Cl)=O)C1 Cc1cc(C(=O)OCC(c2ccc(O)c(Br)c2)C)ccc1OC(F)(F)F Cc1ccc(C)c(CC(=O)NCC2CCCCN2C(=O)C(C)OC(C)(C)C)c1 N1(Cc2c(OC(CC)C)cccc2)CCc2sccc2C1c1cccs1 c1(OC2CC(NC(=O)C(F)C3CC3)C2)cccn2nnnc12.C1(=O)CC(=O)C(C)N1 c1(CCC(N2CC(O)(CC)C2)=O)cccc(NC(C2CCCOC2)=O)n1 c1(C(N2CCC(OC)(CNC(c3ccoc3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 C=CC(C)(CC)C(=O)NCc1cn(C2CN(C(=O)CSCC(F)F)C2)nn1 N1(C(CN(C(=O)OCC)C)=O)CCC(NC(=O)CCC2CCCCN2C)C(C)C1 c1(C(=O)NC2CC2)cc(Cl)ccc1OCCNC(C1(CC)CC1C)=O.C1(=O)CN1 c1(C(=O)OC)ccc(C)nc1NC1CCN(C(c2cc(C)no2)=O)C1C CC1CCCCN1C(=O)C=CC(C)NC(=O)C(CO)N(C)C N1(C(c2cccc(CSC)c2)=O)CC(NC(=O)COC2CCCC2)CC(O)C1 C#Cc1cccc(NC(C2CC(NC(c3cc(F)ccc3C)=O)C2)=O)c1 c1(CNC(C(C)(C2CC2)OC)=O)ccccc1CN(C)C(c1c(C)cnn1C)=O Cc1cnncc1CC(N1CCOCC1c1cn(CCOCCC(C)C)nn1)=O c1(C(N2C(C)CCN(C(=O)C(F)OC(F)(F)F)CC2)=O)c[nH]c2cc(F)ccc12 Cc1nc2ccccn2c1C(=O)NC(C)(CNC(=O)C(C)C(C)(F)F)C1CCC1 N1(C(C(C(=O)OC)C)=O)CCC2CCN(C(=O)C(C)(C)COCC(F)F)CC12 c1(C(=O)NC2CCCN(C(C(C)(C)CC#N)=O)CC2F)cccc2ccncc12 c1(CC)cc(C(=O)NC2CC(CO)N(C(C3CCC(=O)O3)=O)C2)ncn1 Cc1ccc(-c2cccc(-c3cn(C(C)C(=O)NC(C)CF)nn3)c2)cc1 c1(C(=O)NCCC2CCN(C(CNC=O)=O)C2)cc(Cl)c(F)c(Cl)c1 CC1CN(S(=O)(=O)N2CCC(CO)CC2)CCO1.C(N)=O C12(C(=O)NCC3C(CC)CCN3C(=O)CC(F)(F)F)CCCC(CO1)C2 C1(C2CCC2)(CNC(C=Cc2cn(C)nc2)=O)CCN(C(c2cscn2)=O)CC1 C12(CN(c3ccc(CC)c(O)c3)C(=O)CC(=O)OC)CCCC1OCC2 Cc1nn(CC(N2CC(C)CCC2CNC(=O)CC(C)C)=O)c(C)c1Cl C1(CC(=O)N(C(C)(C)C)C2CC2)CCN(S(=O)(=O)CCc2ccno2)CC1 N1(C(C2CC(=O)NC2)=O)CCC2CCCC12C(=O)NCC(O)C1(Cl)CC1 C1(C(=O)NC2CCCN(C(c3cnn(CC)c3Cl)=O)C2)CCc2[nH]nc(O)c2C1 c1(OC(C)C)ccc(C(C2CCCO2)NCc2ccc(F)cc2)cc1 c1(C(=O)NC2CC3(C(C(=O)NC(C(=O)OCC)C)C3)C2)cnc(C)nc1C C1(NC(C2(OC)CCCC2)=O)C2CN(C(c3ccc(C(C)C)nc3)=O)CC12 N1(CC)CCC(CNC(C2C=CC(C(=O)NC(C3CCCCC3)C)C2)=O)CC1 c1(C(=O)NCC2C(C(=O)OC)CCC2)ccc(-c2ncco2)cc1F c1(C(=O)NC(CC)CNC(=O)CCC2CCC(=O)N2)cncc2[nH]ccc12 C(=O)(C(F)(F)CC(C)C)NCC(CC=C)NC(=O)Cc1nnc(C)o1 C(=O)(C(CC(=O)O)N1CCOC(CCN2CCCC2=O)C1)NC(=O)OC(C)(C)C C1(CCOC)CC(O)(C2CCN(C(=O)Nc3nc(C#N)c(C#N)nc3C)CC2)C1 c1(NC(C2SCCN(c3c(F)cnc(OCC)n3)C2)=O)c(Cl)c(F)nc(F)c1Cl c1(NC(c2nc(-c3c(C)ccc(OC)c3)sc2C)=O)ccc2scnc2c1 n1(CC(=O)NC2(C(F)F)CC(NC(C(C)(C)OC)=O)C2)c(O)nc2ccccc12 C1(NC(C(C)N(C(C)=O)C)=O)CCN(C(=O)Cc2cncc(F)c2)C12CC2 Cc1nc(Cl)ccc1CC(N1CCN(C(=O)CC2CCCOCC2)C(CO)C1)=O O(NC(=O)C(CC(N)=O)NC(=O)C(N)=O)CC1CO1.C(C)(C)OCCO Cc1ccccc1C(=O)N(CCCN(C(=O)CCC1CC12CC2)C)C C1(CC(C)CNC(=O)C#CC2CC2)CCN(C(c2ccoc2)=O)CC1 c1(NC(=O)CC2CCCN(C(=O)CC3CCOC3=O)C2)cccc(F)c1F CCC(C(=O)NC1CC(CNC(c2cncn2C)=O)C1)N(C)C C12(NC(c3c(Cl)cncc3Cl)=O)CCCC1N(C(=O)CC1CC1)CCC2 c1(C(N2CC3C(CNC(C(CC)=CC)=O)(C3)C2)=O)cc(C)c(Cl)c(C)c1 C1(C(N2C(C(=O)Nc3cc(O)nc(O)n3)CC(O)C2)=O)CCc2nc[nH]c2C1 c1(N2CC3(C(NC(C4CC45CC5)=O)CCS3)C2)c(Cl)cncc1[N+](=O)[O-] CC1CN(C(c2cc(Cl)no2)=O)CCC1CNC(=O)CCCCN(C)C N1(C(C2C(C(C)C)N(C(c3cnc(S)nc3)=O)CC2)=O)CC(O)CC1(C)C C(=O)(C(=O)C(F)(F)F)NCCC1CCN(C(C(C)CC2CCC2)=O)CC1 c1(C(=O)NCC2(O)CCN(C(c3c(C)nns3)=O)C2)cc(S(N)(=O)=O)oc1C c1(C(=O)NC2CC(NC(=O)C=CCF)C2)cnn(CCC(F)(F)F)c1 C1(C(N(CCNC(C2(OC(C)C)CCSC2)=O)CC)=O)CCn2c(O)nnc2C1 C1(NC(C2=CC(C)(C)C2)=O)CCCC2CN(C(c3ccc(N)cn3)=O)CC12 C12(NC(C(CC)NC(C)=O)=O)CCC(C1)N(C(c1ccc(F)cc1O)=O)C2 c1(NC(CCCC(C)NC(=O)CCc2cn[nH]c2)=O)ccc2cccnc2c1 N1(C(c2cc(C)sn2)=O)CC(C(=O)Nc2cccnc2CO)C(C2CC2)C1 C1(C(=O)NC(CC)CN(C)C(c2cnn(CC3CC3)c2)=O)COCC2(CCC2)O1 C#CC1(O)CCN(C(C2CC(C)CCN2C(c2coc(C)c2)=O)=O)C1 c1(CC)ccc(C(=O)NCCC(C)(C)NC(C2CNC(=O)O2)=O)c(N)c1 c1(C(=O)NC(CC)(CNC(C2(CCOC)CCC2)=O)CC)ccc(F)c(C)c1N N1(C(c2nc(COC)oc2)=O)CC(F)(F)CC1CNC(=O)C(C)C(C)(C)C c1(NC(CC(=O)OCC)C(F)(F)F)cccc2[nH]nc(C3CC3)c12 c1(C(=O)NC(C2CN(C(=O)C(F)CC3CCC3)C2)C)cc(Cl)ccc1F CC(C)CCCC(C)C(=O)N(C1CN(C(C2COC(=O)C2)=O)CC1(C)C)C c1(CC)ncc(Cl)cn1.C1(c2ncno2)CNCCN1 O=C1NCC2(CCN(C(=O)CC3(NC(C4CC(O)C4)=O)CCCCC3)C2)O1 N1(CCOCC)CCC(N=c2[nH]c(=N)[nH]c(=NCCCn3cccn3)[nH]2)CC1 N1(C(COCCCC#C)=O)CCCC(NC(C2CCOC(CC)C2)=O)C1 C1(CNC(C2=NOC(C)C2)=O)CN(C(c2cc(Cl)ns2)=O)C2COCC2O1 N#Cc1cn(CC(N2CCCC23CCN(C(=O)C2=CCCC2)C3)=O)c(=O)nc1O c1(CN2CCC(CC)C2)cc(Cl)ccc1C.C1C(=O)N1CC(C)C C(=O)(C(C)C(F)(F)C(F)F)N1CCC(CCNC(C2(CC#C)CCOCC2)=O)C1 C1(NC(c2c(CCC)nns2)=O)CCN(C(c2ccccc2)=O)CC1CC N1(C(C(c2cnn(C)c2)OC)=O)CC(C)CCC1CNC(=O)C=CBr c1(C(=O)OC(C)(C)C)cn(CC(c2cc(C3CCOC3)[nH]n2)=O)nn1.C1C(=O)O1 c1(COC)nc(C(=O)NC2(C)CC(NC(c3snnc3C3CC3)=O)C2)cs1 C(c1ccc(OCCOC)cc1)=CC(=O)NCCCCC(C)NC(C1C(=C)C1)=O c1(C(=O)NC(CNC(C(C)NC(C2CCCC2)=O)=O)C2CC2)ncc(F)cc1N C(=O)(CS(=O)(=O)CC(=O)NCC1CC(CNC(C23COCC2C3)=O)C1)OC N1(C(c2c(C)nn(C)c2)=O)CCCC(C)C1CNC(C1(c2ccccc2)CC1)=O C1(NC(c2n(CC)ccn2)=O)C(CNC(=O)C(C)=CC2CC2)CCC12CCC2 c1(OC)sc(C(=O)NCC2CC2CNC(c2ccnc(C)c2)=O)cc1Br N1(C(c2[nH]cc(CC)c2)=O)CCCCC(NC(=O)C(C)SC(F)(F)F)C1 c1(C(=O)NCc2c(C)cccc2)csc2c1CCN(C(=O)C(C)(C)F)C2 C1(NC(c2nc[nH]c3nccc2-3)=O)CCCCCN(C(=O)C2=CCOC2)C1 c1(C(=O)NCC(C)NC(C2C(COC)C2)=O)ccc(F)c(N)c1 c1(CNC(C2CCC(CC)O2)=O)ncccc1CNC(c1cnccc1C)=O N1(c2nc(=NC)[nH]c(=NCc3ncc(C)cn3)[nH]2)CCOc2ccc(Br)cc2C1 N1(C(CNS(C)(=O)=O)=O)CCOC2(CCCN(C(C3CCC=CO3)=O)C2)C1 Cc1cc(=NC(=O)C2CCN(Cc3cc(Br)cc(I)c3)CC2O)[nH]c(Cl)n1 Cc1ncc(CC(=O)NCC2CCCN2C)s1.C12(CC1)C(=O)NC2 C(=O)(CCC1=CCCCC1)N1CC(C#C)(C(N2CCc3c[nH]nc3C2)=O)C1 C(CCCCC(=O)NCC1CC(NC(c2ncc(Cl)cc2F)=O)CC1O)SC S(=O)(=O)(c1ccc(C#N)cc1Cl)N1CC2N(C(C(=O)N(C)C)=O)C(COC2)C1 c1(C(N(C)CC2N(C(C3C(=C)C3)=O)CCOC2)=O)cc(C)c(Br)cn1 CC1C(C)N(C(=O)CC2CCCC2)CCN1C(=O)CCc1cc(Cl)cc(Cl)c1 C1(N(C(=O)CC2(OC)CCC2)CC)CN(C(c2cc(=O)cc[nH]2)=O)CC12CC2 C1(C2(C(=O)NCC(C=C)(F)F)CC2)COCCN1C(=O)CC(=O)N(C)C C(=O)(CCCCBr)NC1(NC(COCC(C)C)=O)CCC1 c1(OC)ccc(O)cc1NC(C1(C(C)NC(c2csc(Cl)n2)=O)CC1)=O c1(NC(C2CC2NC(c2cc(C(C)C)cc(F)c2)=O)=O)ccc([N+](=O)[O-])cc1F CCC(CN(C)C)CC(=O)N1CC(C)(NC(c2cnc(C3CCOC3)s2)=O)C1 C(C(C(=O)NCCC(F)F)NC(=O)C(n1ccnc1C)C)SCC C1(C(C(=O)NC2(CC=C)CCN(c3nnc(CC)s3)C2)C)CCC(C)(C)CC1 N1(C(c2cc(C)n(C)n2)=O)CC2CN(C(C3CCN(S(C)(=O)=O)C3)=O)CCC12 CC(C(=O)NCC1CC2CCC1N2C(c1cc(C(F)F)ccc1F)=O)C(C)(F)F C(=O)(C(C)CC(F)F)N1CCC(C(CNC(c2c(C)coc2)=O)C)CC1 C1(N=c2ccc(C#N)n[nH]2)(CNC(C2OCC(C)C2)=O)CCC1 c1(C(=O)NC(c2cccc(C)c2)CNC(c2occc2F)=O)ccc(F)cc1C c1(CC(=O)NCCCN2CCN(C(C)C)CC2)ccc(C#N)cc1 C1(NC(C2C(C)(C)C2)=O)COCCN(C(=O)C(c2ccccc2)=O)C1 c1(COC(c2cccc(C(N)=O)c2)=O)cc(Cl)cc(F)c1O Cc1cc2c(C(N3CCCC(CO)(NC(c4cnns4)=O)C3)=O)ccc(C)c2[nH]1 C1(C(=O)NCC=C2CN(C(C3(C4CC4)CCCO3)=O)C2)COC2(CCC2)C1 c1ccc2c(c1)COC2.C1(CC(COC)OC)CCCCN1C(=O)OC(C)(C)C c1(CNC(C=CCC)=O)nocc1C(=O)NC(C)CC(N)=O C1(C(=O)NCCCCNC(c2ncc(Br)cn2)=O)CCCC(F)(F)C1 N1(CC)CCC(O)C(C)(CO)C1.c12cc(Br)ccc1-c1c[nH]nc1NC(=O)NC2 C1(CC(=O)NC2(CNC(c3cnn(C)c3N)=O)CCOC2)CCC(C)(C)CO1 c1(C(CC)C)ccc(C#N)c(N2CCC(N(C(=O)C(C)Cc3ccco3)C)C2)n1 c1(C(=O)OCC)ccccc1C(C)(C)NC(C1CC1CNC(=O)CC1(C)CC1)=O N1(C(C(C)NC(=O)C2CC2)=O)CCC(CO)C(NC(=O)C=CC2CCCN2C)C1 CS(=O)CCC(O)C(=O)NC1CN(C(=O)Cn2nc3c(n2)CCCC3)C1 N1(C(c2c(C)scn2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C2(CCC2)C1 CS(=O)(=O)c1cccc(S(=O)(=O)N2CC(O)CC2CO)c1 CC1(NC(c2cccc(Cn3cc(C(C)(C)OC(=N)O)nn3)c2)=O)CCNC1=O C1(C)(C(=O)NCC2C(CC)CN(C(C3(C)OCCO3)=O)CC2)CC(C)OC(C)C1 C1(C(=O)NCC2(C3CC3)CCCO2)CC=CCC1C(=O)Nc1ccccn1 N1(C(c2ccsn2)=O)CCN(C(=O)C=CC2CCCO2)CC(CO)C1 C(=O)(CCCCCC#N)NCC(C(N1CCCC(C)(O)C1)=O)OC c1(C(=O)O)cccc(Cn2nnnc2C2(NCC3CCSCC3)CCC2)c1 Cc1nc(CC(=O)N(CC(O)CN(C(=O)CN(c2ccccc2)C)C)C)cs1 c1(C(=O)NCC2CC(NC(C=CC(=O)OC)=O)C2(C)C)cc(Br)c2c(c1)OCO2 C1(C(=O)NC(C(=O)NC2CCC=CCCC2)CC2CC2)Cc2ccccc2C1 O=C(C(O)C(F)(F)F)NCc1cccc(-c2cn[nH]c2)c1 N1(C(C(C2CC=CCC2)NC(CC=CC)=O)=O)CCCC(CO)CC1 Cc1noc2ccc(C(=O)Nc3cc(C(N4CCCC(C#N)C4)=O)n(C)c3)cc12 C1(NC(C=CC=CCC)=O)CCN(C(=O)C(C)(C)C)CC1CO c1(C(C(=O)NCC(=C)C)N(C)CCC2(C)OCCO2)nc(Br)cs1 C1(CNC(CN(CC(=O)NC(C)C)C)=O)COC2COCC12.C12(C)CCCN1C2=O CC1CCN(C(=O)Cn2cc(C3CCOC3)cn2)C(C)C1NC(=O)C=CC(N)=O C(=O)(CCS(=O)(=O)N(C)C)NCCC(C)NC(=O)C(C)OC1CCCCC1 CCC(C)C(O)C(=O)NCc1cccc(C(N2CCCC2)C)c1 c1(NCc2c(C(=O)OC)cccn2)cc(F)c(Cl)cc1F.N12CC(F)(C1)C2=O Cc1nc(N2CCCC(C)(CNC(=O)CC34CCC(CC3)C4)C2)nc(O)c1C Cc1nc2c([nH]1)CC(NC(c1c[nH]nc1-c1ccccc1Br)=O)CC2 Cc1c[nH]c(NC(C2CCCN(C(C3CC3C)=O)CC2)=O)c1C#N c1(CC2CC3CCC2CC3)cc(Br)cc(Cl)c1F.N1(C2C(=O)N2)CCCC1 C(C)(C(CC(=O)NCC1CCOC1C)NC(C1CCC1C(C)(C)C)=O)OC N1(C(COC(CC)(C)C)=O)CC(N(C(=O)CN2CCC(O)CC2)C)C(O)C1 C(=O)(CCC(N)=O)NCC1(NC(c2n(COC)ncc2)=O)CCOC1 N1(CCOCC)CCC(CN2CCN(c3ccc(Cl)cn3)CC2)C(C)C1 c1(C(=O)NC(CN(C(=O)C=CS(C)=O)CCOC)C)ccc2c(c1)CCC2(F)F N1(C(c2c(OC)scc2)=O)CC2(NC(C3OCCC3C)=O)CCCC2(F)C1 C1(CN(C(=O)C(N2CCCC(F)CC2)=O)C2CC2)CCC2(CCCCCC2)O1 N1(C(CC2(CNC(CCC)=O)CC2)=O)CCC(CC2CC2)C1 CS(=O)c1ccc(C(=O)NC2CC(NC(c3ccc(N)c(Cl)n3)=O)C2)cc1 C=C(F)C1(CC(N2CCN(CC(=O)NCc3n[nH]cc3C)CC2)=O)CCC1 C(=O)(C(F)(F)C(C)(C)O)NCC12OCC(NC(C(CC)NC(N)=O)=O)(C1)C2 c1(OCC(=O)NC2C(NC(c3ccc(C)cn3)=O)CCC2)ccccc1[N+](=O)[O-] N1(C(C(C(C)C)F)=O)CC(NC(=O)C=CSNCc2ccco2)CC1(C)C c1(CC(=O)N(CC(CNC(C(CC)C)=O)(C)C)C)c[nH]c2cc(F)ccc12 c1(C2(OC(C3CC(C(F)C(=O)NC(C)(C)C)C3)=O)CC2)ccc(O)cc1 C1(C)(C(=O)NCC(n2cc(C3(C)CCCC3)nn2)C)CCCS1 N1(C(=O)Cc2cc[nH]n2)CC2CCC1C1CN(CCC3CC3)CC21 Cc1cc(C(=O)NCC2CC(F)(CNC(=O)C(C)Oc3cccnc3)C2)sn1 c1(C(N2CCN(C(C)C)CC23CC3)=O)ccc2oc(O)nc2n1 c1(C(N(CCNC(c2cc(CCC)[nH]n2)=O)C)=O)cn2ccc(C)c(C)c2n1 Cc1cc(C(=O)NCC(C)CC(=O)NC2CC3CC3C2)nc(O)c1 n1(CCC(=O)NCCN(C(=O)CC2CCC3CC23)C)cc([N+](=O)[O-])cn1 N(C(=NCCC(C)C)NC1COCC1F)CCc1ccc(OC)c(F)c1 c1(C(=O)NCCC2CC(OC)CN2C(c2coc(Cl)n2)=O)cc(C)c(C)c(F)c1 C=CCCCCCC(=O)N1CCN(C(=O)CC(=O)CCCCO)CC(CO)C1 N1(CCCC=C)CC2CN(C(=O)C(=O)NC3CC3)CC2C1.c12ccc(c(C)c1)o2 N1(Cc2cccc(C)c2)C2CCC1CC(O)(C(=O)Nc1nccc(C(C)C)n1)C2 c1(OC)ccccc1NCC(=O)N(CC(C)NC(=O)Cc1sc(SC)nc1C)C C1(C)(NC(C(C)Oc2ccc(O)cc2)=O)CCCN(C(=O)CCP(C)(C)=O)C1 C1(NC(C=Cc2scc(C)n2)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)CC1 CC1=C(C)CC(C)(NC(=O)CNC(c2ccc(C#N)n2C)=O)CC1 C(=O)(CC(C)C(C)(C)C)N1CCC(C=C)(C(=O)NCC(c2cnc[nH]2)C)C1 C1(C2CCN(C(=O)Cc3c(C)noc3C)C2)(NC(c2cc(CC)c(C)s2)=O)CC1 N(C(=NC)N1CCC(OCC(F)(F)F)CC1)SCC.C12CC(C1)C2 C1(CNC(C(C2CC2)OCC)=O)CN(c2ncncc2OCC(CC)CC)CC(C)(C)O1 CC(C)CC(O)CC(=O)NC(C)(CNC(=O)Cn1cnc(C(N)=O)n1)CO Cc1cc(F)sc1C(=O)NC(C)CNC(C1CC12CCC2)=O CC(C)C(O)C(=O)NCCOCC(C)Oc1ccc(C2CC2)cc1 c1(C(C(=O)CCNC(=O)CC2CCCCC2)=O)cccc(N)c1.NC(=O)CN CS(=O)(=O)N=S1(=O)CCN(C(C23CC(CN)(C2)OC32COC2)=O)CC1 C1(c2ccc(C)cc2)NC(=O)N(CCC(=O)N(c2nnnn2C)C2CCC2)C1=O C(=O)(CC(C(F)(F)F)NC(=O)OC(C)(C)C)NCC(CC)NC(CSC)=O c1(C(=O)NC2C(OC)CCC2)ccc(CNC(=O)CC2CCCCO2)cc1 C12(C(=O)NCC3(CNC(c4c(C)ncs4)=O)CC3)CC=CC(C1)OC2 CC1CCN(C(=O)Cc2cccc3c2CCO3)C(C)C1NC(C12CC1C2)=O C1(C(=O)NCC(CNC(c2cc(C)c(Br)o2)=O)C)C2CCC1(C)C2(C)C c1(C(=O)NC(CC)(CNC(c2cc(C)cc(C)n2)=O)CC)cc(C)nc(Cl)c1N C1(c2nnnn2Cc2ccccc2)(NCc2c(COC)cns2)CCCC(C)C1 C=C(C)C(CC(=O)N(C1CCCC1)CCCNC(=O)CS(N)(=O)=O)OCC.C(COC)O CN(CCCC(=O)N1CCC(C)(CCNC(c2cc3ccccc3s2)=O)C1)N=O C1(CCOC)(NC(=O)CC2COC(C)(C)C2)CCN(C(C2(O)CCOC2)=O)C1 CC(F)(F)C(F)(F)CC(=O)N1CCN(C(=O)CC2CCCCC2)CC1CO N1(C(C2CC(F)CN2C(c2cc(F)c(F)c(Cl)c2)=O)=O)Cc2ccc(F)cc2C1 C1(CC(=O)NCC(CC)NC(c2ccc(OC)c(C)c2)=O)CCCC2(CCC2)O1 c1(C(=O)NCC23C(CN(C(C=CC(CC)C)=O)C2)C3)cc(N)c(Cl)cn1 N1(C(C2(CC)CCC2)=O)CC(NC(c2cc(N)ccc2Cl)=O)C2(CC2)C1 N1(C(C2(CCNC(C(C)C)=O)CCCO2)=O)CCC(C)(CN(C)C)C1 C1(NC(=O)CC2CC3CCC2CC3)CCN(CC(=O)N2CCC2)CC(O)C1 CC(CCN=c1ccc(Br)c(S(=O)(=O)NCC)[nH]1)N(CC(O)C1CCC1)C.N(C)C O=C(C1=C2CCN=C2NC=C1)NC(C1CCCCC1)CNC(C1CC1c1ccno1)=O C1(C)(C(=O)NCC2(C(=O)NC(C#C)CC3CCC3)CC(=C)C2)CCCC1O N(C1CCCc2occc21)C(C1CCCCN(C(C(CCC=C)(C)C)=O)C1)=O N1(C(c2cc(C)[nH]c2)=O)CCCC(C(=O)NCCc2cc(C)[nH]n2)CC1 C(=O)(C1=C(C#N)CCC1)N(CCC)CCNC(=O)C(c1ccc(F)cc1)(F)F C1(C(N(CCC(C)NC(c2sccc2Cl)=O)C)=O)Cc2c(F)cccc2O1 C1(NC(=O)CC2CCC(=O)O2)(Cc2nn[nH]n2)CCCCC1 N1(C(C(CC)Nc2nc(C)cs2)=O)CCC(C2CN(C(=O)CCCF)C2)CC1 Cc1c(C(F)(F)F)cc(C(N2CCN(C3CCOC3)CC2)=O)cc1[N+](=O)[O-] C1(NC(CNC(C(CC)C)=O)=O)CCCN(C(C2CCSC2)=O)C1C Cc1cc(NC(=O)C(c2ccc(F)cc2)NC(N)=O)cnc1C c1(C(=O)NC2C(CNC(CCC(C)OC)=O)CC2)sc(C#N)cc1Cl N1(C(C(C)OCCOC)=O)CCCC(CO)(NC(=O)C(C)c2cccs2)C1 c1(CN2CCCN(C)CCC2)nc(=NCC2CC23CC3)[nH]c2ccsc12 c1(C(=O)OC)cnn(C(C)(C)C)c1Cl.C12COC(C1)CNC(=O)C(=O)N2 C1(C(CNC(COCCN(C)C)=O)(C)C)CCN(C(C2CCCC2OC)=O)CC1 c1(C(=O)OCC)c(N2CCCC(NC(=O)C(C)C3CCCO3)C2)cc(C)nc1O CCCCC(=O)C(=O)N(CCCN(C(=O)C(C)c1cc[nH]n1)C)C N1(C(=O)OC(C)(C)C)CC2CC(OC(=O)C(C)(O)C3CC3)C(C2)C1 c1(C(=O)NCC(N2CCCC(NC(C3(SC)CC3)=O)C2)=O)ccsc1[N+](=O)[O-] N1(C(c2cc(C)oc2C)=O)CC2CCC1C(CNC(C1CC1F)=O)C2 C12(CC(=O)N(C(C)CN(C)C(c3cccn3C)=O)C)CC3CC(C1)CC(O)(C3)C2 c1(CNC2(CC(=O)NC(c3ccccc3F)C)CCC2)ccc2[nH]ccc2c1 Cc1cc(C)c(CC(=O)NCCC2CC(NC(=O)COc3cccnc3)C2)s1 C1(c2cn(CCC3CN(C(C4OCC(C)C4)=O)C3)nn2)CCCC(F)(F)C1 CCC(CCC(=O)NCCn1cc(C(=O)NCCNC(=O)CC)cn1)OC N1(C(c2c(OC)cnnc2)=O)CCCC(CC(N2CCC2C)=O)CC1 NS(=O)(=O)CCCC(=O)NC1CCCC1NC(c1cc2c(s1)CCCC2)=O CCC(CC(=O)NCC(C1CC1)NC(C1(C)CCCN1C)=O)C1CCC1 Cc1cn(C)cc1C(=O)NC1(C(=O)N(C(C(N)=O)C2CC2)C)CC1C Cn1[nH]c(-c2ccccc2)nc1=NC(=O)NC1CCN(c2cnc(Cl)cn2)CC1 N1(C(CC2(C)OCCO2)=O)CCC(CO)(NC(=O)Cc2cc(C3CC3)no2)C1 Cc1ccc(-n2ccc(C(N3CCN(CCN(C)C(=O)C4CC4)CC3)=O)n2)cc1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)Cn2ncnn2)c2c(c1)CCO2 CCC(C)C(c1nnnn1CCOC1CC1)NCCOCC.C1(O)CCCCC1 c1(CC)cccc2c(F)c(C(N3CC4C(NC(=O)C=C(Cl)Cl)C4C3)=O)[nH]c12 Cc1ccc(Cl)cc1C(=O)NC1(CNC(C2CCN(CC(C)C)C2)=O)CCCC1 N1(C(C=C(C)c2ccc(F)cc2)=O)CCCC(C2CCN(C(=O)C=C3CC3)C2)C1 c1(C(=O)NCC(CC)(C)NC(c2ccon2)=O)n[nH]c(C2CC2)c1Br C=CCCC(C(=O)NCC(CC)(CC)OC)NC(=O)C(O)CC1CCCC1 c1(CNC(CC)=O)ccc(C2CCN(C(=O)CCCCNC(N)=O)CC2)cc1F N1(C(c2ncc(C)nc2)=O)CCC(CNC(=O)CN(C)C(N)=O)C(C)C1 C1(C(N(CC(C)NC(c2ccc(SCC)cc2)=O)CC)=O)CCCCC(F)(F)C1 c1(C(N2CCC(F)(CNC(C3(CF)CCC3)=O)C2)=O)cccnc1F C=CCCCC(C)(C)C(=O)N1CC(C(N2CCC(C)CC2C)=O)C(CC)C1 C1(C)(CNC(=O)CC2CCCC2OCC(=O)OC)COCCN(Cc2cncs2)C1 c1(CN(CC2N(C(C=COCC)=O)CCCC2)CC)ccc2ccccc2c1 C(=O)(CC(F)(F)C(C)C)N1CC(C(C)C)N(C(c2nnn(C)n2)=O)CC1 C1(C(C)NC(c2ccc(C3CCCCC3)o2)=O)CN(C(c2ccsc2)=O)CCO1 CC(CS(C)(=O)=O)C(=O)N1CCOC(CNc2ncn(C)c(=O)c2Br)C1 c1(C(=O)NC2CC(N(C)C(C3CC4(CSC4)C3)=O)C2)nnc2ccccc2c1N C1(CNC(COCCCOC)=O)CN(C(c2ccccc2OC)=O)CCN1C c1(C(N2CC(NC(CC3(C)CC3(F)F)=O)C2)=O)ccc(C(=O)CF)cc1 c1(C(N2CCC(OC(C)C)C2)=O)cc(CNC(=O)C=CC(=O)N(C)C)nn1C c1(C(N(CC(C)N(C(=O)CC2CCN(C)C2=O)C)C)=O)cc2n(n1)CCC2 Cc1nc(N2CC3CCCC(NC(C4CC(C(C)C)C4)=O)C3C2)ccc1[N+](=O)[O-] N1(C(CN(C(C(C)C)=O)C)=O)CCC2CN(C(=O)CN3CCN(C)C(=O)C3)C2C1 C1(C(N(OCC(=O)OC)C)=O)CC(NC(c2cc(OC)n[nH]2)=O)CCO1 CC1(C)COCC1C(=O)NC1CN(C(C2CC3CCC(C2)C3)=O)CC1CC1CC1 CCC(C)(CNC(C1CCC(=O)O1)=O)C(=O)NCc1nnc(C)o1 C1(CNC(C2CN(C(C3C4CCC(F)C34)=O)CCO2)=O)CC2(CCC2)C1 c1(OC)cc(C(N2CCC(F)(CNC(=O)C=Cc3nc(C)co3)C2)=O)c(F)cn1 c1(OC)ccc(C2CCN(C(=O)CC3(c4ccc(F)cc4)CC3)CC2)nc1 CCC(CC(F)F)C(=O)NCC1CN(C(=O)CC(C)C(=O)OC)CC(C)(C)O1 C(CC(C)N=c1[nH]c(C(C)C)nc2[nH]ccc12)NC(c1c(C)ccnc1)=O C1(C(=O)NC2CC(CC(=O)NC(CC(C)O)C)C2)CCC(C)(C)OC1 c1(C(=O)NCC(C2CCC2)NC(C(C)C#N)=O)nc(C(F)(F)F)n2ccccc12 Cc1cc(C)c(CC(=O)NCCC(C)N(C(=O)CCC(F)F)C)c(C)c1 C1(C(=O)NC2CC(C)(CNC(c3cnc(C(C)=O)s3)=O)C2)CCOC(=O)CC1 Cc1cccc(CC(=O)NC(C)CCNC(C2(S(C)(=O)=O)CC2)=O)c1Br Cc1ncc2n1CCC(C(=O)NC(C)CNC(C1CC1C(C)O)=O)C2 N1(Cc2ccc(C#N)cn2)C2CCC1CC(NC(c1ccc(I)c(F)c1F)=O)C2 c1(C(N)=O)cccc2[nH]nc(-c3ccccc3O)c12.N12CC3(CC3C1=O)C2 N1(C(CC(C)=C(C)C)=O)CCOC(CN(C(=O)C(C)C2CCCC2)C)C1 C(=O)(CCCCCC(=O)N(CCCNC(=O)Cc1ncoc1C)C1CC1)OCC C(CC(C(C)(C)C)NC(C1CC1c1ccco1)=O)N(C(C(C=C)(C)C)=O)C C1(=CC(=O)N(CC(C)NC(=O)CSCCN(C)C)C)CC2CCC(C1)N2C C(CCC)(C(=O)NC1CCC(OC)C1)OC(CC)(C)C.C1=CCNC1=O C(=O)(C1CCCc2n[nH]cc21)N(CC(C)CNC(=O)Cc1cccnc1Cl)C c1(NC(CN2CCN(Cc3c(C)nn(C)c3Cl)CC2=O)=O)nc2ccccn2n1 Cc1nc(C)c(C(=O)N(CC(=O)N(CC(O)CN(C)C)C)CC2CC2)o1 c1(C(=O)OC)ccc(N2CCC(NC(=O)C3=COCCC3)C(O)C2)c([N+](=O)[O-])c1 C=CCC(CC)C(=O)NC1CC12CC(C(=O)Nc1cc(OC)cc(F)c1)C2 c1(OC)ncccc1N(C)C(=O)CSc1cccc[n+]1[O-] c1(C(C(=O)NCCCCNC(C2CC(=C)C2)=O)=O)cc(Br)cs1 CCC(C)C(O)CC(=O)NC1(CNC(=O)CNS(=O)(=O)c2cccnc2)CCC1 CC1C2CCN1C(=O)COC2=O.N1(C(=O)ON)CCCCC1CO.c1(O)ccccc1 CN1C(=O)C(F)CC1C(=O)NC1CN(C(c2cc(C#N)cs2)=O)CC1O c1(C(N(CC#C)CC2CC2)=O)occc1CNC(c1cccs1)=O N1(C(CCCCCCC)=O)CCC2(CC1)CC(NC(C1C3CCC13)=O)CO2 c1(C(N2CC3(N(C(c4cccc(C)c4)=O)CC3)C2)=O)cc(F)cc(Br)c1F C(C(=O)N1CC(C2CC2)(OC)C1)(C(C)(C)C)NC(C(COCC)C)=O CC(CCC(=O)N1CCC(CNC(=O)Cc2cncnc2)C12CC2)S(C)(=O)=O C1(C)(CC)CN(C(c2[nH]cnc2C)C(=O)Nc2ccc(F)cc2C)CCO1 CCCC(C(=O)N1CCN(CC(C)NC(c2cn(CC)nn2)=O)CC1)NC(N)=O C1(CNC(CCCC(C)=O)=O)COC(C)(C)CN1C(=O)CC1CCOC1=O C(C(O)C(=O)N(C(C)Cn1cc(CN(C)C)nn1)C)=C.CCO N1(C(CC2N(C(CNC(CN(C)C)=O)=O)C3C2CCC3)=O)CC(O)(C2CCC2)C1 C(=O)(C(CC1CCCC1)NC(=O)CC(C)N(C)C)N(CC(C)N(C(C)=O)C)C c1(C(=O)NCCCn2cc(-c3ccc(F)cc3Br)nn2)ccnc2ncnn12 N1(C(C)=O)CC(C(=O)NC2(OC3CN(C(=O)CC#N)C3)CCOC2)C(C)C1 N1(C(C(c2ccoc2)NC(=O)CC2CC=CCC2)=O)CCC(O)CC12CC2 CC1(C)CCCCCC1S(=O)(=O)Cc1cccc(OCCS(N)(=O)=O)c1 Cc1cnc(C(N2CCOCC2CNC(=O)CCS(C)(=O)=O)=O)c(C)c1 N1(C(CCCOC)=O)CCCC(CO)(CNC(=O)CCC2(C)CC2(F)F)C1 C1(NC(c2cscn2)=O)CC2CCC1CN(C(=O)C1CCCc3ncnn31)C2 N1(C(C(C2CCCCC2)C)=O)CC2CC(NC(c3ccc(Cl)s3)=O)CC1C2 c1(OC)cnc[nH]c1=NCC1CCCC(NC(C2CCN(C)C2=O)=O)C1 C(=O)(C(C)(C)C(=O)N1CCCCC1CNC(c1csc(C)n1)=O)NC n1(C(C)C)nnc2c1C(C(=O)NC1CCC1)CN(Cc1ccc(Br)cc1F)C2 Cc1cc2nc(NC(=O)C(=O)Nc3ccc(=N)[nH]n3)sc2cc1C O=C(C1CCc2ccccc21)NCC1CCCCN1c1nc2c(F)cccc2o1 c1(N(C)Cc2cccc(F)c2)nc(NCCn2cnnc2)c2ccsc2n1 n1(CC(=O)NCC2CC(NC(C(CCCC)O)=O)C2)ncc2ncccc12 N1(C(CNC(C)=O)=O)CCCC2(CCCN2C(=O)CCc2ccccn2)C1 C(C(F)(F)C(=O)N1COC(C)C1)Oc1ccc(SC)cc1 N1(C(c2c(C)cn(C)n2)=O)CC2CC1CCC2NC(=O)Cc1c[nH]nc1C Cc1cnc(C(N2CC(NC(C3CC4(CC4)CO3)=O)CC23CCC3)=O)cc1C#N N1(C(C(C)Cc2ccc(Br)cc2)=O)CCOC2C(C(F)(F)F)CC12.C1C(=O)O1 c1(C(=O)NC2CN(C(C(C(=O)OCC)F)=O)CC2SC)nc2ncc(C)cn2n1 N1(c2nnc(CC)o2)CCC2C(CCCN2C(c2cccnc2)=O)C1 C1(NC(C(C)OC)=O)COC2(C1)CN(C(c1c(N)cccc1F)=O)C2 N1(C(C)C)CCOC(C(=O)NCCCC2CN(C(c3cc(F)n[nH]3)=O)CCO2)C1 C1(CC)CCN(C(=O)C(F)C(C)CNC(c2ccc(CO)o2)=O)CCO1 Cc1ccc(CC(N2CCN(CCCNC(=O)C(C)N(C)C)CC2)=O)cn1 c1(OC)ccc(C2C(C(=O)OCC(=O)Nc3nccs3)C2)cc1OC C1(NC(c2cc(C)n(C)n2)=O)CC2CC(NC(c3cnc(Cl)c(N)c3)=O)C1C2 C(=O)(C(C)C(C)COC)NC1CC(NC(c2n[nH]c(CC)c2Br)=O)C1 Cn1cnc(=N)n1C(c1coc(-c2ccccc2)n1)C1CC1 Cc1cccc2c(C(=O)NC(C3CCCN3C(c3c[nH]ccc3=O)=O)C)coc12 C(=O)(CC1=CCCCC1)NCC(CNC(c1coc(C(C)C)n1)=O)OC Cc1ccc(NC(C2CN(C(=O)C(C)(C)Br)CCC2O)=O)cc1F Cc1cc(C)nc(N2CC(NC(c3cn(CC4CCCOC4)nn3)=O)CC2C)n1 N1(C(c2cccc3[nH]ncc23)C(=O)NC(CC)(C)C)CC2CC3CC2C1C3O C1(CC(=O)NCc2ccc(C(=O)NC(CSC)(C)C)o2)CCC(C)(C)O1 C1(NC(C(C)NC(N)=O)=O)C2CC3CN(C(C4CCCC4(C)C)=O)C1C3C2 c1(C(=O)NC2C(C)N(C(=O)CC3CC3(C)C)CC2)c(Cl)c([N+](=O)[O-])nn1C C1(NC(c2cnc(C(C)C)s2)=O)CC2CC1CN2C(c1ccccc1C(F)F)=O CCCCN=C(NCCN1CCCC1)NCC1(C)CCC(C)CC1 C(=O)(C(CC(C)(C)C)NC(=O)CC1CC(C)C1)N1CC(CC(C#C)C)C1 C1(NC(C(N2CCSCC2)C)=O)CN(C(=O)COCc2ccccn2)CC1(C)C C1(N=c2[nH]nc(C(F)F)o2)(CCC)CCN(C(=O)C(CC=C)CC(F)F)CC1 C(CC1=CCCCC1)NC(C1CCCN(C(CCSC)C(=O)O)CC1)=O c1(C(N(C2CN(C(C(COC)(C)O)=O)CC2O)CCO)=O)cc(F)ccc1OC C1(NC(c2ccc(CN(CCC)C)o2)=O)CN(C(c2[nH]cnc2C)=O)CC12CC2 c1(C(=O)NC2CCN(C(c3nnc(CC)s3)=O)CC2)cc(C)c(O)c(C)c1 CN1C(=O)CCC1CC(=O)NCc1ncccc1C(N1CCC(C)(F)C1)=O c1(C(=O)NCCOC2CCN(C(CC3CCN(C)C3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl C1(CC(=O)N(C)CC2CCCN(c3nnn(C)n3)C2)CCOC(C)(C)C1 C1(N(C(CC=C)=O)CCOC)CC2(CCNCC2)C1 Cc1cc(C(=O)NCC2CC2NC(=O)CC2(n3cncn3)CC2)cnc1C(F)F C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1(CNC(c2nc(CC)oc2C)=O)CC1 C(CN=c1[nH]cncc1I)(N(C)C(c1nn(C)cc1Cl)=O)C1CC1 C1(NC(C2(CO)CCN(C(C(C)OCC3CC3)=O)C2)=O)C(C)(C)C(O)C1(C)C C1(C2CCN(C(=O)CCCCCC#N)C2)(NC(CN(C(C)=O)C)=O)CC1 C(=O)(CCCC(C)=O)N1C(C(=O)NCC2(F)CCCCC2)(COC)C=CC1 c1(OCC)cccc(C(=O)NC2CCC(CNC(=O)CNC=O)C2)c1N C1(COC)CN(C(c2ncc(C(C)(C)C)cn2)C(=O)NCCCSC)C(C)(C)C1 C(C1(O)CCc2ccccc21)N(C(C=C)C1CCC1)C c1(NC(C(N2C(c3cc(C)[nH]n3)CSCC2)=O)=O)cccc(F)c1[N+](=O)[O-] C1(CC(=O)NC(C2(CNC(=O)CCc3cnoc3)CC2)C)CCOCC1 CC1CN(C(=O)CCC2(C)CN(C(C3CCN(C)CC3)=O)C2)CC1(F)F CC1COc2c(C(=O)NC(C)CC(C)NC(=O)CN(C)C)cccc21 CC1(C)C=C(C(=O)N2CC(OC(C3(C(C)(C)O)CC3)=O)C2)C1 c1(CNc2c(C(N(CCOCC)CCO)=O)scc2)cc(Br)ncc1Br C12(C(N(CCNC(C3(CCOC)CCC3)=O)C3CC3)=O)CCC(CC1)C2 c1(C(=O)NC2CCC2NC(c2cc[n+]([O-])cc2)=O)coc2c1C(=O)NCCC2 C1(C(=O)NC2(CSC)CCC2)CCN(C(c2cnnc(O)c2)=O)CCO1 C1(OC)CC(CNC(c2n[nH]cc2C)=O)N(C(C2CCN(C)C2=O)=O)C1 C12CN(CC(=O)N1)C2=O.C1(NC(=O)C(C)c2cccs2)C2CCC1CNC2.CO c1(OC)cccc(CCC(=O)NC(C)CC(C)NC(c2ccsn2)=O)c1F N1(C(Cc2ccc(C)c(C)c2)=O)CCC2CN(C(c3nc(Br)cs3)=O)CC2C1 C1(NC(C(C)OC)=O)CCC2CC1CN2C(c1c(Cl)n[nH]c1C)=O c1(C(C=CC(=O)N(C(CCC)C)CC)=O)ccc(Cl)cc1 C1(C)(NC(C(CNC(C2N(CC)CCC2)=O)N(C)C)=O)CC(C)(C)C1 C1(NC(CC2(C)N(C(c3cc(C)cc(O)n3)=O)CCC2)=O)CCn2nnnc2C1 c1(C(=O)NCC(CC(C)C)NC(C(C(CC)O)C)=O)nc(N)cc2ccccc12 CC1(NC(=O)CNC=O)CN(C(=O)C(C2CC2)NC(=O)CCCCO)CCO1 C1(NC(C2CCN(C)C2)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC2(CC2)C1 C1(C(=O)NCC(CSC)(C)C)C2CCC(C2)N1C(=O)C(C1CCCCC1)C c1(NC(C2C(C(=O)NCc3cccc4cc[nH]c34)C2)=O)c(Cl)cc(Cl)cc1Br C#CCCCCCC(=O)N(C(C)CN(C)C(c1cc(F)cc(N)c1F)=O)C N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2(CCCCC2NC(C2CC2(C)C)=O)C1 N1(C(CC)=O)CCCC12CCN(C(c1cc(C)c(C(=O)OC)o1)=O)C2 c1(N2CCCC(C(C)NC(c3c(C)nns3)=O)C2)nc(Cl)nc2ccc(Cl)nc12 c1(CNC2C(C)(C)CN(C(=O)CCC(F)(F)F)C2)ccc([N+](=O)[O-])cc1F N1(C(C(n2c(C)cc(C)n2)C)=O)CC(NC(=O)CC2OCCO2)CC12CCC2 C1(NC(CC(CC)C2CCC2)=O)CCN(C(C2(O)CCCCCC2)=O)CC1CO Cc1cc(C(N2CCOC(C(=O)NC(C)C#N)C2)=O)c(F)cc1F C1(C2(Oc3ccccc3)CC2)CN(C(=O)COCC)CC1c1c(CC)cccc1 c1(C(=O)NCCN(CCOC)C(C2CC2C)=O)cccc(OC(F)F)c1 O=C(CCCC(=O)C1CC1)NCc1cc(C(=O)NCc2ccns2)on1 C1(C(=O)NC2CN(C(=O)CC3CNC(=O)O3)CC2C)(CC)CCCC1O C#CCC(C)(C)C(=O)NCCN1CCCN(C(c2cc(CCOC)on2)=O)CC1 Cc1ccc(F)c(CC(N2CCC(C)(NC(C3CC34CC4)=O)CC2)=O)c1 c1(C(=O)NCCOC2CCN(C(CC3(C)CCCO3)=O)C2)cc(Cl)ccc1C(F)F Cc1cc(C(=O)NC2CC(NC(=O)Cc3cc(C)on3)C2)c(C)cn1 CC#CCCCC(=O)NC(CC)CCC(=O)NC(C)(C)C(=O)NC N1(C(c2cnc(C(C)O)s2)=O)CCOC(CNC(=O)C=Cc2cnc[nH]2)C1 Nc1cc(F)cnc1C(N1CC2CCC2(C(=O)NCc2nc(O)cc(O)n2)C1)=O C1(COCC)CN(C(C2CC(=O)N(Cc3ccccc3Br)C2)=O)CCO1 CC1(C)CCCC(C(=O)NCC2CN(C(c3ccnc(F)c3N)=O)C2)CC1 C1(n2cc(COC)nn2)(C(=O)N(C(C)C(C2CCCO2)=O)C)CCOCC1 c1(C(C(=O)NC2CC2)N(C(c2ccccc2)CC)C)cc(C)nc(C)c1 C(=O)(CCCC1CCC1)NC(CNC(C(C)OC1CCCC1)=O)(C)C1CCC1 C1(C(=O)NCCCN(CC)CC)(Cc2nc[nH]n2)CCCC1.C1(=O)CN1 C(C)(C(=O)N1CC(NC(=O)C(C)(C)CO)CC(F)C1)(C(C)C)OC N1(C(CCC2CCCN(C(c3cc(C)sc3N)=O)C2)=O)CCC(C(N)=O)C1(C)C c1(C(C)=O)nc(C(=O)N(C(C)CNC(=O)C(C)(c2ccccc2)N(C)C)C)cs1 CCC(C)C(C(=O)NC)N(C=O)Cc1cncc(OC)c1 N1(C(c2c(CC)nco2)=O)CC(CNC(=O)CC2CCCS2(=O)=O)C2(CCC2)C1 Cc1cc(=O)oc(C)c1C(N1CC2CC1C2NC(C1CN(C)CC1C)=O)=O C1(O)(CNC(=O)CCc2cn[nH]c2)CCN(C(c2ccccc2C(F)(F)F)=O)C1 C1(OC)CC2(C1)CN(C(=O)CNC(=O)C(F)CC1CCC1)C2 C(C(C)(C)CC(=O)NCC(C)N(C)C(c1cnc(C2CC2)s1)=O)OC(C)=O N1(C(C(C(C)C)(C)C)=O)CC(NC(=O)CC2(C)CC2(F)F)CCC(O)C1 c1(OC(C(=COC(C)C)C#N)=O)cc(Oc2ccccc2)cc(F)c1 c1(C(=O)NC(CC)CNC(c2c(C)nn(C)c2C(F)F)=O)nn(C)c2c1CCC2 c1(C(N2CC(C)(NC(=O)CC3CCCCO3)C2)=O)csc2nnsc12 N1(C(C2CC(=O)NCC2)=O)CCN(C(c2cccc3ncnn23)=O)CC(O)C1 N1(C(CC=C(C)C)=O)CC=C(C(C)(C)C(=O)N2CCCC(O)C2)C1 c1(CC)cc(C)c(C(N2CC(NC(c3ccnn3C3CCC3)=O)C3CC23)=O)o1 N1(Cc2ncc(C)s2)CCC(C(=O)NC2(N(C)C)CCCC2)C(O)C1 c1(C(=O)NC2(C)CCCN(C(C3=C(C)CCC3)=O)C2)n[nH]c2c1CCSC2 C1(C(=O)NC2CCN(C(C(C)OCCOC)=O)CC2C)CCC(C2CC2)CC1 c1(SC)ccccc1C(N1CC(CCCCNC(C2CN(C)CCO2)=O)C1)=O N1(C(C2C(NC(C(C)=CC3CC3)=O)CCC2)=O)CCOC(C)(C(C)C)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C(C)C)NC(C1CCC(C(C)C)O1)=O Cc1cccc2cc(C(=O)NCC3CCCN3C(c3cc(Cl)ncc3N)=O)sc12 CCC(O)C(=O)N1CCC(C(=O)NC2CSC2)C1 c1(S)ccc([N+](=O)[O-])c(N)c1.c1(C(=O)OC(C)(C)C)cn(CC2CCOC2)nn1 c1(CC)ccc(C)cc1NC(=O)C(O)C(C)(C)NC(=O)OC(C)(C)C N1(C(C)=O)CCN(CC(C)F)CC1.c1(NC=O)nccc(-c2ccccc2)n1 c1(C(N2CC3CN(C(C(CCC)CC)=O)C3CC2)=O)c[nH]c2cccc(F)c12 C1(C(=O)NCCCC2CN(C(C3(F)CC3)=O)CCO2)CC2(C1)CC21CC1 N1(C(CCCC)=O)CCC2(CCOCC2)C(CNC(=O)CCCCC(F)F)C1 C1(CNC(c2ccc(Cl)nn2)=O)CCN(Cc2cc(Cl)c(O)cc2F)CC1(F)F C(=O)(C1=Cc2ccccc2C1)N1CC(C(=O)NCC(COC)(F)F)CC12CCC2 CC1C(NC(=O)CCc2ccc(Br)s2)CCCN1C(=O)COC(F)F C1(C(N2CCC3(CC3C(=O)N(C)CC3CC3)C2)=O)CCn2ccnc2C1 Cn1cc2ccc(C(N3CCC4(C3)CN(C(c3ncccn3)=O)C4)=O)cc2n1 CC(F)CC(=O)NC(C1CCCCC1)CNC(=O)CNc1ccccn1 c1(C(C(=O)NC(CC)C)N(CCOC)CCN(C)C)ccn(CCCC#N)n1 CC1CCC2(CC1)CCC(C(=O)NCC1CNC(=O)N1c1ccccc1)O2 c1(C(N(CCCNC(=O)C=Cc2ccc[nH]2)CC)=O)cc2cccn2c(O)n1 C#CCC(C)C(=O)NCCCNC(c1ccoc1Br)=O c1(N2C(CCCNC(C(C)NC(COC)=O)=O)CCC2)nc(Cl)nc2[nH]cnc12 c1(C(C(=O)NCCCSC)N(CC)Cc2ncoc2C)nocc1C1CC1 N1(CCCn2cc(COC(=O)CNc3cccc(N)c3)nn2)CC2COCC2C1 CN1CCOC(C(=O)NCC2(F)CC(NC(=O)CS(C)(=O)=O)C2)C1=O C1(N(C)CC)COCCN(C(=O)C(C)OCCCNC(C)=O)C1 CN1CCOc2cc(CNCC3(C(=O)Nc4cc(F)nc(F)c4)CC3)ccc21 c1(C(=O)NCC2C(NC(C3(C=C)CC3)=O)CCC2)cc(CC)oc1C CON=Cc1ccc(C(=O)NCC2(F)CN(C(=O)C#CC3CCOCC3)C2)cc1 C(=O)(C#CC1CCCCC1)NCC1CCN(C(C(C=C)C)=O)CC1O Nc1cc(C(=O)NC2CCC2NC(c2n[nH]cc2Cl)=O)c2ccccc2c1 N1(C(Cc2ccc(C)cc2)=O)CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1 C1(C(N2CCCC(C(=O)NC(c3c(C)n[nH]c3)C)C2)=O)CC(=O)CC(=O)N1 c1(OC)cccnc1C(=O)NCCC1(O)CN(C(C2OCCC2C(F)(F)F)=O)C1 N1(C(CC(CC)OC)=O)CC(NC(C2CCc3ccnn3C2)=O)CC12CCC2 c1(C(=O)NCC(CC)(C)NC(=O)CCCCCC#N)ccc2[nH]c(C)c(C)c2c1 c1(C(N2CC(F)(CNC(CC3C(OC)COCC3)=O)C2)=O)cc(C)nc(Cl)c1N c1(CCCC(=O)Nc2c(OC)cccc2)ccc(Cl)c(Cl)c1.C1C(=O)N1CC(C)O CC(C)(C)CCC(F)C(=O)NC1CC(NC(C2COC2)=O)C1 N1(C(C(C)NC(=O)C2CC2)=O)C2CCC1CC(CCNC(=O)C(O)C(F)(F)F)C2 C1(O)(CCNC(C(C)CO)=O)CCN(C(=O)Cc2cncnc2O)C1 c1(C(=O)NC2C(C)CN(C(c3ccncc3F)=O)C2)ccc2nnnn2c1 C1(NC(C2CCC2)=O)CCN(C(c2ccc(CC3CCCC3)cc2)=O)CC1 C(CC(=O)N=c1ccn(C(C)CC)[nH]1)C1CC(NC(C(CC)=CC)=O)C1 CCC(C)(C(=O)N1CC2CCC1CN2C(=O)C=C1CCCCC1(C)C)C(N)=O C12(NC(CCCCC)=O)CCCC(CN(C(c3cccc4sncc34)=O)C1)C2 N1(C(C(C(C)C)NC(C)C)=O)CC2CCC1C(NC(C1(O)CC1)=O)C2 C=CC(C)(CCOC)C(=O)NCCOCCCN(C)C(c1cccnn1)=O c1(OC(C)C(=O)NCC(F)CNC(=O)CC2CC=CC2)ccc(Cl)cc1Cl C1(C(=O)NCCC2CC(NC(CC3(OC)CC3)=O)C2)CNC(=O)CC12CCOC2 c1(OCCC)ccc(C(=O)NCCC2CCCN2C(C2CC2(C)C)=O)cc1 C(=O)(C(C)(C)C(=O)NCC(C)N(C(=O)CC1CC1(Cl)Cl)C)OCC C1(NC(C(c2ccnn2C)C)=O)CCC(NC(c2cn(C(C)(C)C)nn2)=O)CC1 n1(CC)cc(C(=O)NC2CC(CNC(C3CCC(OC(F)(F)F)C3)=O)C2)c(C)n1 CCC(CNC(=O)C(C(C)O)NC(=O)C=CC1CC1)C(C)(F)F c1(CC(N2CC(CNC(c3c(OC)noc3C)=O)C(O)C2)=O)cc(C)cc(C)c1 C(=O)(CS(=O)(=O)c1ccccc1C)NC1CC(NC(CC2CC(CC)OCC2)=O)C1 c1(CNC(C2(CNC(CC(C=C)C)=O)CC2)=O)ccnc2[nH]ccc12 C(=O)(C(COC)C(C)C)NC(CC=C)C(=O)NCCSCC=C Cc1nc2[nH][nH]cc-2c(=NC2CCC3CN(C(=O)C(F)(F)C(C)(C)O)CC23)n1 CC(C)(O)C#CC(=O)NCc1nocc1C(=O)NCc1cnn[nH]1 C1(NC(C(CCC)OC)=O)(CO)CCCN(C(c2c(C)nnn2C)=O)C1 C1(O)(C(=O)OC)CC2(CCOCC2)C1.c1(CC)noc(C)c1CNC(=O)NC c12cccc(F)c1N2.N1(C(c2ccncn2)=O)CCC2(CC1)CC2 c1(OC)cc(C(=O)N(C)CC2(O)CN(C(=O)C(O)CN3CCCC3)C2)ccc1C N1(C(C(=O)OC)=O)CCC(OCCNC(c2sccc2C)=O)C1 c1(-c2cccc(CNC(c3cccc(F)c3Br)=O)n2)c(O)cccc1O N1(C(c2c(C)c[nH]n2)=O)CC2(CCCN(C(=O)CCc3ccc(CO)cc3)C2)C1 N1(C(c2ccc(COC(C)C)cc2)=O)CCC(O)(CNC(=O)C(C)O)CC1 C1(C(=O)NCCC#CC)CCN(C(=O)C(CO)NC(N)=O)C(C)C1 N1(C(c2ncc(OC)nc2)=O)CCCCC(C(=O)NC(C)C(C)SC)C1 c1(C(=O)NCC2CCC(NC(CC3(C)CCC3)=O)C2)cnn2c1NCCC2 C1(CNC(C(C(C)C)CO)=O)CN(c2ncc(F)cn2)CC2(CCC2)C1 NC(=O)CCCCC(=O)N1CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C(=O)(C(O)CCC(C)C)NCC1CC1CC(=O)NCc1ncc(C)[nH]1 c1(C(N2CCN(C(CCC=C)=O)C(C)CC2)=O)ccc(C#N)c(F)c1Br Cn1cc(S(=O)(=O)NC2CCC3(CC2)OCCO3)ccc1=O N1(C(c2cc(CC)c(CC)o2)=O)Cc2nccn2CC(NC(C2CC2(Cl)Cl)=O)C1 CC(C)CC(C)(O)c1cn(CC(=O)NC2CCCN(C(C)C)C2)nn1 N1(Cc2cn(CC(CNC(C#CCN(C(C)C)C)=O)(C)C)nn2)C(=O)CNC1=O c1(C(N2CC(N(C(C(C(C)C)n3cnnc3)=O)C)C2)=O)cc(F)cc2nn[nH]c12 C(=O)(C(C)(C)C(C)C)N1CCC(CC=C)(NC(=O)C=Cc2ccc(C)s2)C1 S(=O)(=O)(c1ccccc1F)N1C(CNS(c2c(C(=O)O)ncs2)(=O)=O)CC(O)C1 N1(CCCOc2ccccc2-n2ccnc2)CCC2(CC1)CNCCO2 Nc1ccc(F)c(F)c1C(N1CC(NC(=O)Cc2cnns2)CCC(O)C1)=O Cc1sc(Br)cc1C(=O)NCC(CNC(C1CCS(=O)CC1)=O)CO C1(C(N(CC(C)NC(c2cnnn2C)=O)CC)=O)CC2(CCCC2)CO1 c1(NC(C2CCCCN2CC2CC3C=CC2C3)=O)cccc(C2CC2)n1 Cc1c(CN2CCN(C(=O)NC3CCCCC3)CC2)cc(Cl)cc1Cl CC(CC(C)(C)O)C(=O)OC1CCCOC1.N1(C2(C)CNC2)CCN(C)CC1 C#CCC(C)(C(=O)N1CC(O)CC1(C)CO)NC(=O)Cc1ccc(F)nc1 N1(C(=O)CC2CC23CC3)CC(F)(C2C(CNC(=O)C(F)(F)c3cncs3)C2)C1 N1(C(CSCCCC)=O)CC2CC2(CNC(C2CC2F)=O)C1 CC(C)(Cc1cn(Cc2cccc(Br)c2)nn1)C(=O)N1CCCC1F Cc1cccc(C(=O)NC2CC2CNC(c2cncc(N(C)C)c2)=O)c1C S(=O)(=O)(c1cccc(F)c1)NC(C(C(C)C)N(C1CC1)C1CC1)=O C1(CC)CC(C(=O)N(C)CC2CCN(C(=O)CSC)CC2)CCO1 N1(C(c2ccncc2Cl)=O)CC2CCC1CN2c1nc(Cl)ncc1F CCC(CC)C(C(=O)N(C)CC1COCCN1C(C1OCCCO1)=O)OC c1(CC)ccc(NC(N2CCC(O)(CNC(=O)C(F)=C3CCC3)C2)=O)cc1 C1(O)(C(=O)NC2CC3CC2N(C(=O)CC2CCCC2)C3)CC2(CCOCC2)C1 c1(NC2CC(F)(CNC(C3CCCC(C)C3)=O)C2)ncc2c(c1C#N)CCC2 C(C(C)(O)CC(=O)NCCCCCCn1cc(C2CCCC2O)nn1)OC CC1CC(NC(c2cc(OCC(F)F)ccn2)=O)CN1C(c1cccn1C)=O C1(CC)CCC(C(N2CCOC(CNC(=O)C(O)CSC)C2)=O)CC1 C1(N(c2cnc(C)nc2C)CCc2nn(CC)nc2C)COC2(CCNCC2)C1 N1(C(Cc2c(C)ccc(F)c2)=O)CC(C2CN(C(=O)CC3CCC(=O)C3)C2)C1 C=C=C(C)CC(=O)NC1(C2CCCCN2C(=O)CCN2CCCC2=O)CC1 C(=O)(CC1=NNC(=O)C1)N1CCC(CNC(CCc2cccc(C)c2)=O)C12CC2 CC1CN(C(=O)C(C2(C)CC2)NC(C2CCC2C)=O)C(C)C(C)(C)O1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC2C(NC(C3CC3[N+](=O)[O-])=O)(CCC2)C1 C(=O)(NNc1cc(Br)ccc1F)N1C(Cc2cccc(OC)c2)CN(C)CC1 c1(OC(C)C(=O)NC2CC2CNC(C2CC(C)(C)C2)=O)cccc(Cl)c1Cl c1(CNC2CC3CC(CC(=O)OC)C2C3)c(C)cc(CN)cc1C C1(CC(=O)NCC2CC(O)CN2C(c2ccc(OC)o2)=O)(CC)CCOCC1 C1(CC)CN(C(=O)CC(F)(F)F)CCN1c1ccnc(Br)n1 C=CC(C)(C)N1CC(C(CC2CC2)NC(=O)OCC)C1.C(C)(C)(C)O c1(C(N(CCCCNC(C2C(C)(C(C)C)C2)=O)C)=O)cnnc(C2CC2)c1 CCC(CC(=O)NCCCc1cccs1)N(C(=O)C(CSC)OC)C c1(SCc2cncc(C)n2)ccc(C(=O)NCC(N2CCOCC2)=O)c(C)n1 c1(NC(C(CC)NC(C2C3CCC(C3)C2C)=O)=O)cccc2c1OCO2 C(=O)(C1=CCS(=O)(=O)C1)N1CC2(CC(NC(=O)C(F)CC3CCCCC3)C2)C1 C(=O)(CCCCCN(C(c1ncc(Cl)cc1Br)C(=O)NCC(F)F)C)OC CN1C(=O)OCC1C(=O)NCCC1CC(C(=O)N(c2ccsc2)CCO)C1 c1(N2C(C)CC(CC(C)Nc3ccc4cncn4c3)C2)ncc2cccnc2n1 Cc1cc(C)c(C(=O)NCC2COCCN2C(c2cnc(O)n2C)=O)s1 CC(C)(Cc1ccccc1)C(c1nnnn1CC(F)F)NCC1(C)CSCCO1 Cn1c([N+](=O)[O-])cnc1NC(=O)CSc1ccc(F)cc1 Cc1ccncc1C=CC(=O)NC(C1(O)CN(C(C2CC3CC3CC2C)=O)C1)C N1(C(C(C)Oc2ccccc2F)=O)CCN(C(=O)Cc2csc(=N)[nH]2)CC(O)C1 c1(CC)cccnc1C(N1CCC(C(=O)NC2C=C(C)CCC2)C1)=O C#Cc1ccc(C(=O)NCC2(C3(O)CN(C(C4CC4OCC)=O)C3)CC2)cc1 C(C)(N=c1nc2sccc2c(NC2CN(C(C)C)C2)[nH]1)c1c(COC)cccc1 c1(C(N(CC(CN(C(CC(C(=O)OC)C)=O)C)O)C)=O)cnc2cc[nH]c2c1 c1(C(=O)NCCC2N(C(CC(CC)C)=O)CCSC2)ccc(F)cc1C#N c1(C(N2C(C)CCC(NC(C3C(OCC)C3)=O)C2)=O)cccn2nccc12 c1(C(=O)NC2CN(C(C3CNC(=O)O3)=O)C(CO)C2)cc2ncsc2[nH]1 c1(C(C)C)cccc(F)c1C(=O)NCCNC(=O)Cc1ccco1 C1(C(NOCC=C)=O)(CNC(c2cc(Cl)ns2)=O)CCCO1 C1(NC(COCCC=C)=O)CCN(C(=O)COc2ncccc2CC)CC1C C1(OCC)CN(C(=O)OC(C)(C)C)C(C)(CO)C1.C(C)(C)(CCC=C)O C(C)(C)(CCCN=c1ccnc(SC)[nH]1)NC(c1c(Cl)nc(CCCC)s1)=O CCCCC(O)CC(=O)N1CCC(F)(CNC(=O)CCc2cc[nH]n2)C1 c1(CC(C(=O)NC(C(CO)NC(C2(C(CC)=O)CC2)=O)C)C)ccccc1C c1(C(=O)NCC(CNC(c2cc(Cl)cc(C)c2N)=O)O)ccc2c(c1)CCC=C2 CCC(C)CC(C)C(=O)N1CCC(CCNC(C2CC(C)(C)C2)=O)CC1 c1(C(N2C(C(=O)Nc3cc(OC)ncc3)CCCC2)=O)ccn2cncc2c1 Cc1cc(N)c(C(N2CCC(OC3CN(C(C4C(C)C4C)=O)C3)CC2)=O)cc1C CCCC(C(F)(F)F)NC(C1CCCN(C(c2cc(C)nn2CCC)=O)CC1)=O C1(C#N)(CN(C)C)CCC1.c12cnn(c1)CCSC1CC1NC2=O C1(CNC(CCN(CC)CC)=O)CC2(CC2)CN1C(C1NC(=O)OC1C)=O N1(C(COC)=O)CCC(N(C(=O)CCCNC(c2ccsc2)=O)C)CC1 c1(C(=O)NCCCNC(C=C(C)C2CCCCC2)=O)c(N)sc2ccccc12 Cc1cc(C(=O)NC2CC2NC(C2C=CCC2)=O)c(C)s1 S(=O)(=O)(c1ccc(Cl)cc1F)N1CC(C(=O)NCCc2nc[nH]n2)NCC1 CC1CCc2[nH]nc(C(N3CC4CC(NC(=O)CCCC(N)=O)C3C4)=O)c2C1 C1(C(N(C(C)C(=O)NC(C(N)=O)C2CCCC2)C)=O)CCCN1N1CCCC1 C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1C(NC(CCCCCCC)=O)COC1 C1(C(=O)NC(C(=O)N(C(C)CO)C)Cc2cn[nH]c2)CC(=O)CC1(C)C c1(CC(=O)NCCc2cn(-c3cc(C)cc(N)c3)nn2)cccc2cccnc12 S(=O)(=O)(c1nccs1)NC1CCCN(C(c2cccc(Br)c2F)=O)C1 C1(CC(=O)NC2(C(N3C(C(C)O)CC3)=O)CC2)CC2CCC1O2 C(=O)(CCS(=O)(=O)Cc1ccccn1)N1CCC(OCCNC(=O)C(F)F)CC1 N1(C(C2CC(OC)C2)=O)CC(NC(c2cc3[nH]ccc3s2)=O)CC2(CC2)C1 C12(SCc3cn(CC(=O)NCC(=O)Nc4c(C)n[nH]c4)nn3)CCC(C1)C2(C)C c1(CCNC(c2nnnn2CSc2ccccc2)CSCC)ccc(F)c(Br)c1 N1(C(C)C(=O)NC2CC(CC(=O)NOCCO)C2)CCCCC1.C1(OC)CC1 c1(C(N2CC(NC(C(C)C3CCCO3)=O)(CO)C2)=O)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(C(CCC(N)=O)NC(N)=O)N1CC(N(C(Cc2ccc(C)cc2Cl)=O)C)C1 C=C(C)CN=C(NCC(O)SC1CCOC1)N(C)CC(=O)N(C)C C1(CC)CN(C(c2nn(CC)cc2Cl)=O)CCC1NC(C1CC1C(C)O)=O N1(CC)CC(NC(=O)C(=O)N(Cc2nc(C)no2)CC2CCCCC2)CCC1=O c1(C(=O)NCCC(C(C)C)NC(c2cscn2)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2cc(C)nnc2)=O)CCN(C(=O)CCCCCF)CC1CF C(=O)(CC1=CSC2=NCCN12)NC(CC(C)NC(=O)CCCc1ccc(C)s1)C CC(=O)CC(C)(C)CC(=O)NCC(C)N(C)C(C1CCC(=O)C(C)C1(C)C)=O C12(CC(N3C(C(=O)NC)CC3)=O)CCC1CN(C(=O)CC1CCCCC1)C2 c1(NC(COC)CO)ccc(S(=O)(=O)NCc2c(F)cccc2Cl)c(Cl)c1 C(N=c1[nH]c(=NCC2CCC3(CC2)CC3(F)F)c2ccccc2[nH]1)C1CC(C)C1 CCC(C(=O)NCC1CCCCN(C(=O)C(=O)NC)C1)C(C)(F)F c1(CC(=O)NC2CC(NC(C(C(CC)C)OC)=O)C2)ccc([N+](=O)[O-])c(N)c1 N#CCCCCC(=O)N1CCC(NC(C2CC3CCC2O3)=O)CC1 c1(COCC#C)nc(C)sc1C(=O)OCc1cccc(Br)c1 CCC(C)(C)C(=O)C(=O)NC1CCN(C(c2c(C)noc2C)=O)C1C Cc1cc(NC(=O)CNC(=O)C#CC2CCC2)cnc1Cl c1(C(=O)NC(CNC(CSCC=C)=O)C(C)C)cccc(C)c1N N1(C(C2CCN(CC(C)C)CC2)=O)CCN(C(=O)CC2CC2(C)C)CC(CO)C1 CCCCC(C(=O)NCC1CCCN1C(=O)C(C(C)(C)C)OC)N(C)C c1(C(=O)NC(C2CCCCC2)CNC(=O)CO)cc2n(n1)CCCC2O C(CC(C)C)(C(=O)N1CCC(CF)(NC(=O)CC2CC(=O)C2)C1)OC N12CC3(C(F)(F)F)CC3(C1)C2.CC(C)(C)CCn1cc(C(=O)OC)nn1 O=C1C2CS(=O)(=O)CCN2C(=O)N1Cc1ccccc1OCC(F)F c1(C(=O)NC(C)C(CO)NC(=O)COc2ccsn2)ccn2ncnc2c1 C1(NC(=O)C(F)C2CC2)CC2(C1)CN(C(C1(C3CCCO3)CC1)=O)C2 C1(NC(Cc2nc(C)sc2C)=O)CC(F)(F)CC1NC(c1c(C)nc(C)n1O)=O CN1CCC(C(CCOC)NCC2CCC(NC(c3cc(CO)[nH]n3)=O)C2)CC1=O C(N=c1ncc2[nH]ccc2[nH]1)C1C(N)CCCCC1 c1(N2CCCC(CNC(C#CC(C)(C)C)=O)C2)ccc([N+](=O)[O-])cc1F C(CNC(C12CC(F)(C1)C2)=O)(C(C)(C)C)NC(Cc1cc(C)no1)=O N1(C(C2(C#N)CC2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C2(CCC2)C1 CC(C)CCCC(C)CNC(C1CCC=CC1NC(=O)C(C)c1ccco1)=O c1(NC(c2ccccc2-n2cc(CC3(O)CCC3)nn2)C)nccc(Cl)c1C N1(C(CCCOCCOC)=O)CC2CC(NC(c3ccco3)=O)CC1C2 c1(C(N(C(=O)C=Cc2ccc(Br)s2)C(C)=O)C)ccc(F)cc1 C(CC1=CCCCCC1)NC(CC1CC(NC(C2(CC(C)C)CC2)=O)C1)=O c1(CC(=O)N(C2CCCN(C(c3c(CC)nns3)=O)C2)C)ccc(C#N)cc1 C=C=CCC(=O)NC1COCC1NC(=O)C(F)F c1(C(=O)NC2C(NC(C(C=C)(C)C)=O)CC2)c(F)ccc(C)c1Cl C1(C(N(C2CCN(Cc3noc(C4CCC4)n3)CC2)C)=O)CCCC(F)C1 CC1(C(=O)NCC2(NC(c3cccc(CC(F)(F)F)c3)=O)CCC2)COCCO1 Cn1nc(CNC(=O)NCC2(NC(=O)OC(C)(C)C)CCC2)cc1Br c1(C(=O)NCC2(CNC(C3(C(=O)NC)CC3(F)F)=O)CCC2)c(C)ccc(C)c1O N1(C(C2CCN(C)C2=O)=O)CC2CCCC2(C(N2CCCCC2)=O)C1 Cc1cc(NC2CC2C(F)(F)F)ccc1COCc1ccc(C)c(Cl)c1 c1(C(=O)NCCN(C(=O)COc2ccsn2)C2CCC2)ccn2ccnc2c1 c1(C(N(CCC(=O)NC(C2CCCC2)CC)C)=O)ccc(O)nc1 c1(CC(C(=O)N2CC(N(C(=O)C(N)=O)C)C2)NC(N)=O)ccc(F)cc1 C1(OC(C)(C)C)CC2CC(NC(=O)NC3(C)CC4CCC3C4)CC12 c1(SC)ccc(C(N2CC3C(NC(c4cn5c(n4)SCC5)=O)C3C2)=O)c(Cl)c1 CC1(NC(c2ccncn2)=O)CN(C(C2COCOC2)=O)C1 C(C(O)CC(F)(F)F)NC(C(C(C)NC(c1cccc(CO)n1)=O)C)=O Cc1nc(-c2cn(C3CN(C(=O)CSC4(CCC(F)(F)F)CC4)C3)nn2)sc1C CCCCC(CNC(c1ccc(C(F)(F)F)nn1)=O)NC(C1CC1F)=O c1(C(=O)Nc2ccc(COC)c(Cl)c2)ccc2c(C)c[nH]c2c1 CCCC(CNC(=O)C(C)(C)C(=O)OC)C(=O)NCc1n[nH]c(C)n1 c1(COCC(=O)NCCC2(NC(=O)C(=Cc3c[nH]cn3)F)CCC2)ccccn1 C1(NC(c2ccc(OC)s2)=O)CCCCC1CNC(c1c(C)[nH][nH]c1=N)=O c1(C(N2CCN(Cc3ccc(OC)cc3)CC2)=O)ccnc(Cl)c1OC c1(C(N2C(CCNC(c3c(C)snc3)=O)CCCC2)=O)cc2c([nH]1)CCC(C)C2 c1(C(N2C(CNC(CC)=O)CC(COC)C2)=O)c(Br)ccc(F)c1N C12(C(N3CCC(Nc4nnc(-c5ccon5)s4)C3)=O)CCCC1C2(F)F C1(C(N2CC(C)CC(CC)C2)=O)N(C(=O)C2=NNC(=O)C2)CC12CCCC2 C(C)(CNC(c1ccsc1CC)=O)(CC(C)C)NC(c1cccc(CCC)c1)=O N1(C(c2nc(CNC(C(N3CCOC3=O)C)=O)oc2)=O)CCC2(CC1)N=N2 c1(OCCN(C(=O)Cn2cc(CCO)nn2)C)cc(C(=O)O)c[nH]1 C1(NC(CSCCCCC)=O)C=CC(C(=O)NC(C)CC(C)O)C1 CCC(C)CC(=O)N(CCNC(=O)C(N1CCC(O)CC1)C)C1CC1 c1(C(=O)NCCCCCNC(Cc2c(C)ccs2)=O)c(C(F)(F)F)cncc1F N1(C(C2(CC)CCOCC2)=O)CCC(C)C(NC(c2ccncc2)=O)C1 CCC(CC(=O)N(CC(O)CN(C(=O)C(F)n1ccnc1)C)C)OC C1(NC(C2(CNC(C(CC=C)NC(C)=O)=O)CC3(CC3)C2)=O)CCOC(C)(C)C1 C1(NC(c2nc(C)sc2)=O)CN(C(=O)CCc2ccc(F)nc2)CC2CCCC12 c1(C(=O)NC(C(C)C)CNC(=O)CC2CC=CCC2)ccc2c(=O)cc[nH]c2c1 c1(C(=O)NCCC2CCCN(C(COCCC)=O)C2)ccc(C(C)CC)nc1O C1(=CC(N2CC3C(NC(=O)C=CCn4cncn4)C3C2)=O)CN2CCC1CC2 c1(C(N2CCCC(NC(c3c(N)non3)=O)(CO)C2)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(CC2N(C)CCC2)=O)CCCCN(C(c2cncnc2)=O)CC1 CC(CN(C(=O)C#CC1CCCOC1)C)N=c1ccn2c(Br)cnc2[nH]1 c1(OC)cc(CNC(=NCCCc2cccs2)NC(CF)CF)cc(OC)c1OC CCN(C(C)c1cccc(C)c1)N1CCN(C)CC2(CNC2)C1 N1(CC(N2C(C(C)C)CCCC2)=O)Cc2ccccc2C1=O c1(OC(CN(C(C=C)C)CCNCC)=O)ccccc1COc1ccc(C)cc1 C#CC1(C(=O)NC2CN(C(c3ccncc3Br)=O)CC2C)CCCC1 Cc1noc(Cl)c1CC(=O)NCCN(C(c1conc1CC1CC1)=O)C1CC1 c1(C(=O)NC2(C(=O)NCC=CCCC)CCCC2)cc2ccccc2[nH]1 C1(C(=O)Nc2scc(C(N3C(COC)COCC3)=O)n2)COCCC1(F)F CN1CCC(C(=O)NC(C)(C)CNC(C2NC(=O)C3CC23)=O)c2ccccc21 c1(C(=O)NC2CC(NC(C3CC(O)(CC#C)C3)=O)C2)ccc2ccc(Cl)cc2n1 C=CC1CCCCN1C(=O)C(C(C)(C)C)NC(C1CC(C)N(C)C1)=O c1(C(N(C)CC2N(C(C(CC)O)=O)CCC2)=O)ccc(OCF)cc1 Cc1oc(CNC(=O)CCCC#N)nc1C(N1CCC(CC(C)(C)C)C1)=O Cc1cn(C(C)(C)C(=O)NCC(C)NC(=O)CCc2nncn2C)cn1 C(CC(O)CCO)NC(C(C1CCCC1)NC(=O)CCc1ccccc1)=O c1(C(=O)NCC2CCN2C(=O)C=C(Cl)Cl)ccc(=O)n(CCO)c1 CC(C)(CCCF)C(=O)NC1CC(CNC(C23CCCC2C3(F)F)=O)C(O)C1 [N-]=[N+]=Nc1cc(F)ccc1C(=O)NCCC1=CCN(C(=O)CNC=O)CC1 CC(C)C(N=[N+]=[N-])C(=O)NCC1(NC(=O)CCC2CC2)CCOC1 C(CC(C)C(=O)N1CCCC1C(N1CCCC1CCO)=O)=CC c1(CCC(=O)NCc2ncon2)cccc(F)c1Br.C12(CC)CC(C1)C(=O)NC2 c1(C(N2CCCC(CNC(c3c(OC)scc3)=O)C2)=O)ccc(O)nc1Cl N1(C(C(N)=O)=O)CCC2(C1)CN(C(c1csc3cccc(Br)c13)=O)CCO2 C1(N(C(C2CN(C)C(=O)N2)=O)C)CCC2CN(C(c3csc(O)n3)=O)CC12 c1(COC)ncc(C(N2CCCC(NC(c3n[nH]c(SC)c3Cl)=O)C2)=O)c(O)n1 Cc1cc(C(=O)NCC23CCC(C2)N(C(c2cc(C(F)F)[nH]n2)=O)C3)cc(F)c1 CC(F)(F)C(C)(C)C(=O)NC1CCC(NC(=O)COc2cc(Cl)cc(Cl)c2)C1 CC(C)C1=CCC(NC(=O)CN(CCCc2ccccc2C(F)(F)F)CC)CC1 C1(NC(c2ncn(C)c(=O)c2)=O)(CNC(=O)C=CC(=O)N(C)C)CCC(F)(F)CC1 CCCCCC(C1CC1)OC.c12cccc(c1)CC1CCN(CC1)C2=O n1(CC(=O)NC2(CNC(C3(CCF)CC3)=O)CCCC2)ncn(O)c1=O N12CCC(CC13CC3)NC2=O.c1(C(C)NC(C)C)ncco1 CC1CN(C(=O)Cc2cn(-c3ccn(C)n3)cn2)CC1CNC(=O)CSC1CC1 C(C(=O)O)(C(O)c1cccnc1)NC(C(n1cc(Cl)cn1)C)=O c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cc(C)c(Cl)cc1C N1(C(=O)Nc2ccc(C(=O)OC)s2)CC2(CCC(Nc3cc(C)cc(Cl)c3)C2)C1 c1(C(N(CC(C)N(C(C(C)OCCCCCC)=O)C)C)=O)ccc(Cl)cn1 C=CCCCC(C)(C)C(=O)N1CCN(C(C2OCC3COCCC23)=O)C(CC)C1 C1(C(=O)NC(CC(=O)NC)C)C=CCN(C(c2cn(C)nc2C)=O)C1 Cc1c(C(N2CC(NC(=O)CCN3CCC(O)CC3)C(O)C2)=O)nn(C)c1N C1(c2ccc(CC)cc2)CN(C(C2(SC)CC2)=O)CCN1C(c1coc(Cl)n1)=O C(C)(C)(CC(F)C(=O)NC(C)C(=O)N(C)C1CC1)NC(c1c(CC)cco1)=O c1(SC)c(C)nc2scc(NC(N3CC(NC(=O)OC(C)(C)C)C(C)C3)=O)n12 C(=O)(CC1=CCN(C)CC1)NC(C1CN(C(c2cc(F)c(Cl)cc2Cl)=O)C1)C Cc1ccc(C(C)C)cc1C(N1CCC(C(C)NC(=O)CCCOC(C)C)C1)=O C1(C(=O)NCC(C)NC(=O)CS(=O)(=O)C2CC2)Cc2cc(Cl)ccc2O1 c1(CC)noc(C(N2CCC(O)(CNC(=O)CC3CCC(C)(C)C3)C2)=O)c1C Cc1cccc(C(=O)N(CC(C)C(=O)NCC2CCC(C)C2)C)c1F N1(C(C(C2(O)CCC2)NC(=O)CCCc2ccco2)=O)CC(C2CCCCC2)C1 C1(C(N2CC(OCCN(C)C)C2)=O)CSCCN1C(=O)C(O)CN(C)C c1(C(=O)OCC2CC2C(F)(F)F)cc2ncccn2n1 n1(CC)nc(C(N2CCC(NC(=O)C(C3(O)CCCC3)F)C2C)=O)c(Br)n1 c1(C(=O)NC(C2OCCN(C(C(C)C)=O)C2)C)cc2nc[nH]c2cc1F c1(C(=O)NCC(CC(=O)N(CCN=[N+]=[N-])CC)C2CCC2)ccc([N+](=O)[O-])o1 c1(CC(N2CC3CN(C(c4c(C)c[nH]n4)=O)CC3C2)=O)ccc([N+](=O)[O-])cc1F N1(C(CCSC)C(=O)NC2CCC(F)(F)CC2)CCCC1C1OCCO1 c1(C(N(CCC)CCNC(=O)C=CCF)=O)c(COC)cccc1CC c1(C(N2CC(C(C)NC(=O)C(C)(Cl)Cl)OCC2)=O)ccc(=O)n2c1CCC2 c1(NC(c2ccc(CNC(c3ccc(OC)nc3)=O)cc2)=O)scc(O)c1C#N C#CCCCC(C)C(=O)NC1C2CC1N(C(c1cnc(C3CC3)nc1)=O)C2 c1(C(C(=O)NC(CNC(Cc2nc(C)[nH]n2)=O)CO)(C)O)ccc(F)cc1 CCC(Cc1cccc(F)c1)C(=O)NCC(c1cn(C2CCCC2)nn1)(C)O c1(C(N(C)CC2N(C(CSC)=O)CCC2)=O)ccc2nc(O)n(C3CC3)c2c1 C#CC1(C(=O)N(CC(C)C)CCC)CCN(C(=O)C(C)=CC(C)(C)C)CC1 N1(C(=O)NCC(c2cccc(F)c2)O)CC2(CO)CC(c3ccc(F)cc3)(C1)C2 CC(C)(CNC(=O)C(C1CCOCC1)NC=O)Cn1cc(-c2cc[nH]n2)nn1 CC1(C)CC(NC(=O)C=CCO)CCN(C(C2CC3(CCCC3)CO2)=O)C1 C(=O)(C(C)C(F)(F)C(F)F)N(CCNC(C(C(CC)(C)C)O)=O)C(C)C c1(CC(N2CCN(C(COCCCC)=O)C3C2C3)=O)c[nH]c2c(CC)cccc12 N1(C(C=CC(CC)C)=O)CC2CCC1CN2C(=O)CCCc1ccc(C)c(C)c1 C1(CCC)CN(C(C2CC23CC3)=O)CC1C(=O)CC.C1(N)(COC)CC1 Cc1ccc(O)c(CN2CCCC(C(=O)NCC3(C4CCCO4)CC3)CC2)c1 Nc1c(C(=O)NC(c2ccccc2Cl)CCO)cc(F)cc1Br C#CCCCC(C)C(=O)NCCC(C)(C)NC(c1coc2c1COC2)=O O=C(C#CC1CCCCO1)N1CCN(c2ncnc(O)c2Br)CC1 C(=O)(C1COc2ccc(Cl)cc21)N1CCCC(CN(C(=O)Cc2cccs2)C)C1 c1(N2CCC(C(C)NC(c3cnc(Cl)cn3)=O)C2)nc(C(F)F)nc(=N)[nH]1 C1(NC(=O)C(F)C2CCCC2)CCOC(C(N2CCC3(CC3)C2)=O)C1 C=CC1(C(N2CCC(C(C)C(=O)NCC(C)(C)C3CC3)C2)=O)CCOCC1 c1(C(=O)NC2C(NC(CN3CC(C)C3)=O)C2)ccc(-c2cn[nH]c2)cc1 N1(C(C2C(OC)(OC)CC2)=O)CC(CNC(c2ncoc2C)=O)CC1(C)C CC1CCN(C(=O)CCCc2cnn[nH]2)C(C(=O)NCCCC2CCCCO2)C1 C1(C(=O)NC2C(NC(=O)CCc3ccsc3)C2)CCCC2(CCC2)O1 c1(CCC(=O)NCC2CN(C(=O)Cc3cnoc3)CCO2)cc(F)ccc1F c1(C(=O)OC)ccc(C(=O)N(CC(O)CN(C)C(c2ccc(SC)s2)=O)C)[nH]1 c1(CN(C)CC2(C)CC2(F)F)cc2cc(Cl)ccc2s1 CC(C)CCCN=c1[nH]c(N2CCC3(CCCN(C)C3)C2)nc2ccc(Cl)cc12 c1(OC)cc(CN=c2[nH]c(C(=O)Nc3cn[nH]c3)cs2)ccc1C(C)=O C1(C)(CC)C=C(C(=O)NCC2CN(C)CCN2C(c2csc(C(C)=O)n2)=O)C1 C(C(=O)N(C1CCCN(C(c2c[nH]c(Br)c2)=O)C1)CCO)(C(C)C)OC C=C(C)CC(C(=O)NCCCNC(c1ccc(CC2CC2)s1)=O)NC(C)=O c1(C(=O)NCC2(O)CC(NC(c3c(N)ccc(O)c3)=O)C2)ccnc2c1CCC2 N1(C(C(n2c(C)cc(C)n2)C)=O)CCCC(C)(CNC(=O)CC2(C)CCOC2)C1 N1(CC(=O)N(C2(c3ccc(F)c(Cl)c3)CC2)C(C)C)CCCCC(C(C)(C)C)C1 C12CCCC1(C)C(=O)N(C)C2.C(C(=O)NC1CC1C)NC(=O)OCC C1(OC)CC(C)CN(C(C2(CNC(=O)Cc3ccnc(O)c3)CC2)=O)C1 N1(C(=O)CN2CCOC2=O)CC2(C(N3CCCC(CCO)CC3)=O)CCC1CC2 C1(NC(CNC(c2ccc(C)s2)=O)=O)CC2CN(C(C34CC(C3)C4)=O)CC12 C1(NC(C2N(C)CCC2)=O)CN(C(c2cc(O)ccc2F)=O)C2(CCOCC2)C1 N1(c2snc(CCOC)n2)CCCC(C)(C)C1CNC(=O)CCN1CCCCC1 C1(NC(C(CC)N(C)C)=O)CN(C(c2ccc(CSC)cc2)=O)C(C)(C)C1 N1(C(CC(OCC)OCC)=O)CCC2(CC1)CN(C(C1CC1C)=O)CC2OC C(=O)(C(C#N)CC)NC(CC)CN(C(=O)COCc1ccncc1)C CCC(C(=O)NC1(CO)CCN(C(=O)C(=O)NC)C1)C(=O)NCCOC c1(C(=O)NC2(CN(C(C3(OC)CC3)=O)C)CC2)cccnc1C(F)F N1(C(c2cnc(C)s2)=O)CC2(CCN2C(C2(Oc3ccc(Cl)cc3)CC2)=O)C1 c1(C(=O)NC(C(C(C)C)C)CNC(c2ccc(Cl)cn2)=O)cnc2[nH]ncc2c1 C(C(O)(C(=O)NC1CCCC(NC(C2CC(F)(F)C2)=O)C1)C(F)(F)F)N(C)C C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(C)C2CC2)CC1F c1(C(=O)NCC=CCNC(C(C)SCCCC)=O)csc2cc(OCC)ccc12 C1(NC(Cc2c(C)cccn2)=O)CC(F)CN(C(C2CCC(=O)N2)=O)C1 CC1C(=O)N(C)CCN1C(=O)CCC1(NC(c2ccncc2O)=O)CCC1 C(=O)(C(C)(C)C(=O)NCC(C1CCN(C(c2cnc(O)c(C)c2)=O)CC1)O)NC N1(C(c2c(CC)ncs2)=O)CCCC2CN(C(=O)C(c3ccccc3C)C)CC12 c1(C(=O)NCC2C(NC(COCC=C)=O)CCC2)cc(=O)c2ccccc2n1C C1(NC(C(CC)Oc2ccccc2)=O)CN(C(=O)Cc2nc(C)cs2)CC1SC c1(C(=O)NC2C(NC(C3(C(F)F)CC(=C)C3)=O)CCC2)cc(F)cnc1OC N1(C(C#CCNC(C2CCCCCC2)=O)=O)CCOC2CCCCC12 c1(C(=O)NCCCOCCN(C(C(C2CCCCC2)C)=O)C)cscc1Cl Cc1ncc([N+](=O)[O-])n1CC(=O)Nc1cnn(C2CNC2)n1 CC1=C(C)CC(C(=O)N(CC(C)(C)C(=O)NC2CCN(C(N)=O)CC2)C)CC1 CC1Cc2ccccc2C1NC(C1(c2ccc(N(C)C)cc2)CC1)=O C1(CC(=O)NC(CCOC)C)CCCC(NC(=O)Cc2ncccc2F)C1 c1(C(=O)NC(C2CCN(C(c3c(C)c[nH]n3)=O)C2)(C)C)nn(C(F)F)cc1Cl C(=O)(C(CCC(C)C)CC(=O)OC)N1CCC(F)(CNC(CCC=C)=O)C1 C1(C(N2C(C(=O)NCc3cc(Cl)ccn3)CC=CC2)=O)CC2CCC(C1)O2 N1(C(C(C)(C)OC(C)C)=O)CCN(C(C2(C)CCCS2)=O)CC12CCC2 n1(CC)cc(Cl)c(C(=O)NC(C(C)NC(c2conc2COC)=O)C(C)C)n1 c1(C(=O)NCc2cc(C(N(CC(C)O)CCF)=O)on2)cc2occc2[nH]1 c1(CC(=O)NCCN(C(=O)C2=C(C)CCC2)CC)ccc2ocnc2c1 c1(COC)ccccc1C(=O)NCC(O)CNC(c1cc(C(=O)OC)n[nH]1)=O CC1CC(C(=O)NCC(O)CN(C(=O)CC2CC(F)C2)C)C1 n1(CC)ncc(C(N2CCC2CNC(C2CCCN2C)=O)=O)n1 c1(CC(N2CC(CC(C)NC(c3c(CC)cno3)=O)C2)=O)ccc(F)cc1 c1(C(=O)NC2CN(C(C(CC)C(C)O)=O)CC2(C)C)ccnc2[nH]ncc12 N1(C(c2cnc3n2CCCC3)=O)CCC2(CCCN2C(=O)C2=CCOCC2)C1 N1(C(CSc2ccc(C)cc2)=O)CCn2c(CNC(=O)C=CCF)nnc2C1 C1(NC(c2c(CC)nc(C)o2)=O)CN(C(=O)Cc2ccccc2O)CCC1C C(CCCC(=O)N1CCC(F)(C(=O)N(C2C3CCCC23)C)C1)OC(C)C C1(CNC(c2cnc(COC)s2)=O)CCC(C)CN1C(c1cscc1OC)=O c1(SC)cc(C(=O)NCCC2(O)CCCNC2)cc(SC)c1 N1(C(c2cc(C)ns2)=O)CCN(C(c2ccc(F)s2)=O)C2CCCC12 C1(CCNC(c2cc(OCC)no2)=O)CC(F)(F)CN1C(=O)C(N)=O C1(NC(c2[nH]cc(CC)c2)=O)CC2CC1CN2C(c1nocc1C(C)C)=O C1(C(N2CCCC(CN(C)Cc3ccncc3)C2)=O)CC12CCC(F)(F)CC2 C1(C(N(CC=CC(=O)NC(C(=O)NCC=C)C)C)=O)(OC)CCOC1 C1(CC(=O)NC(CC=C)CNC(c2cnc(CC)nc2)=O)CCCS(=O)(=O)C1 C(=O)(C(C)C(O)C(C)C)NCCN(CC(C)O)C(c1nc(C(C)C)oc1)=O CC1(C)CCC(CC(=O)Nc2cccc(NC(=O)CC3C=CS(=O)(=O)C3)c2)C1 CCC(CC)C(C)C(=O)NCc1cc(C(N2CCCC3C(=O)NCC23)=O)n[nH]1 c1(C(N(C2CC(NC(CC3(CC)COC3)=O)C2)C)=O)nc(C)oc1C N1(C(C(CC(C)C)C)=O)CCCN(C(c2csc(-c3ncc[nH]3)n2)=O)CC(CO)C1 c1(C(=O)NCC2(F)CN(C(C3C(CC)CCC3)=O)C2)cccc(C(C)(F)F)n1 N(C1CCCc2sccc21)C(CCCCCO)c1n(C(C)C)nnn1 C1(C)(CC)CC1C(=O)NCC1CC(C(=O)NCC(C)(C)n2ccnc2)C1 CCC(CC(=O)NCCC1CN(C(c2cc(Br)c[nH]2)=O)CCO1)OC C1(OC)(CNC(C2CC(F)(CO)C2)=O)CCN(C(=O)CC2OCCC2(C)C)C1 C(=O)(C(C#N)C(C)C)NCC(c1ccccc1)NC(c1[nH]cc(C)c1)=O c1(OCC)cnc(C(=O)NC(CNC(=O)CCOC2COC2)CC(C)C)cn1 c1(C(N(CC(CN(C(Cc2c(C)non2)=O)C)O)C)=O)nccnc1N C1(C(=O)OCc2coc(Cc3ccccc3)n2)CNC2(CC2)CO1 CC(C)CC(C(=O)Nc1cc(Cl)cnc1O)NC(=O)C(C)CC#N Cc1c(F)cc(C(=O)NC2CCCCN(C(=O)C=Cc3cscn3)C2)c(F)c1N Cc1ncsc1C=CC(=O)Nc1cccc(NC(=O)C(F)(F)c2cncs2)c1 C1(CC)CCC(C(N2CCC(C(=O)NCc3nc(=O)o[nH]3)C2)=O)O1 N1(C(C(CC)C)=O)CC2(C(=O)NC3CC(n4cncn4)C3)CCC1CC2 N1(C(C(C)=NOCC#N)=O)CCCC(CC(=O)N(C(C)CO)C2CC2)CC1 C(=O)(C(C)(C)CC(=O)N1CC2CCCC2(NC(c2ccoc2C)=O)C1)OCC C#CCCCC(C)C(=O)NCC(C1(O)CN(C(=O)COc2ccc(C)cc2)C1)(C)C c1(C2(C(N3CCC(NC(c4c(CC)c[nH]n4)=O)C3)=O)CC2)cc(F)cc(C#N)c1 c1(-c2ccccc2C)cc2ccccc2s1.c1(NC(CSC)=O)nccs1 c1(C(N2CC(CNC(CSCC=C)=O)C3C2C3)=O)nc(C)ccc1C C1(CC(=O)NCCC(CNC(=O)COCC2CC2)O)CCC(C(N)=O)CC1 N1(C(COCCCC#C)=O)C(CNC(=O)C2=C(Cl)CCOC2)CC2CCCC12 c1(OC)ccc(C(=O)N(CCCN(C)C(C2CC23CCCOC3)=O)C)c(O)c1F C1(C(=O)NCC2(C(C)(C)O)CN(C(Cn3c(C)cnc3)=O)C2)CCCC(C)(C)O1 CCN(OC(=O)C(c1ccccc1)O)C(=O)CNn1ncc(S)c1.CC C1(NC(C=C(CC)CC)=O)CC12CCC(NC(=O)C=C1CCN(C)C1)CC2 Cc1cc(C)c(C(=O)CCCC(=O)OCc2cc(C)ncc2Cl)c(C)c1 O=c1nc2nc(n1C1CCCCC1)NS2.c1(C(O)C2CC2)cc(F)cc(F)c1 N1(C(C(C)C(C)(C)C)=O)CC2CCC1CN2C(C1CCNC(=O)C1)=O c1(C(=O)NCC23N(C(CC(C(=C)C)OCC)=O)CC(C2)C3)cc(C)c(C)c(C)c1 Cn1nc(C2CC2)cc1C(=O)NCC(c1cccc(Cl)c1)NC(C1CCC1(F)F)=O [N-]=[N+]=NCC(C(=O)N1CCS(=N)(=O)CC1)NC(=O)CC1CC2CC2C1 CC1CC(CNC(=O)C2CC2)CN1C(c1ccc(N2CC3CC3C2)cc1)=O c1(OC)ccccc1C(CNC(C1CC1F)=O)NC(c1ncc(F)cn1)=O N1(Cc2ccc(OC)c(O)c2[N+](=O)[O-])CCn2c(nc3ccccc23)C1 CCC(CC(=O)NCC1CC1)CCC1(OCC(=O)NC)CCOCC1.OCC C1(C(N2CC(O)(CN(C(=O)CNC(N)=O)CC)C2)=O)CC(C2CCCC2)C1 c1(C(N(c2ccc(F)cc2)CC)=O)cnc(CNC(=O)CC2CC(F)C2)nc1 C(=O)(CC(C)(O)C(F)(F)F)NC(C)CN(C(=O)C(C)CCc1ccccc1F)C c1(C(=O)NCCN(C(C(c2ccccc2)SC)=O)C)cc2cc(Cl)ccc2s1 c1(CNC(C2(C)CS(=O)(=O)C2)=O)cnn2c1CN(C(C1(C)CCC(=O)N1)=O)CC2 C1(NC(c2cnc(C3CC3)s2)=O)COCCN(C(c2ccccc2Br)=O)C1 c1(C(C)NC)cn(C2CN(C(c3scnc3C3CCCC3)=O)C2)nn1 C1(CNC(CCC2N(C(CCC(=O)N(C)C)=O)CCCC2)=O)CCCCC1(F)F c1(C(=O)NC(C(C)NC(c2csc(S)n2)=O)CO)ccc(Cl)c(Cl)c1 c1(C(=O)NCC=C(C(=O)NCc2c(CC)noc2)C)cccc2cncn12 C#Cc1ccc(C(N2CCSCC2C(=O)Nc2nccnc2Cl)=O)c(Cl)c1 c1(C2(C)OCCO2)ccc(NC(=O)CN2CCOCC2C2CCCCCC2)cc1 C=C(C)CCCC(=O)NCc1nc(C2CCN(C(C3CC3(F)F)=O)CC2)n[nH]1 N1(C(CCc2c(C)n[nH]c2C)=O)CCC2(CCCN2C(c2cnnn2C)=O)CC1 CC(C)C(C)(CNC(C12CCN(CC1)C2)=O)NC(c1cnc(C2CC2)[nH]1)=O CC1CC(=O)NCCN1C(C1C2CN(C(=O)CC(C)(C)O)CC12)=O C1(NC(CC(=O)NCC)=O)CC2CC(C1)N(C(=O)C(c1cc(F)cc(F)c1)C)C2 CN1CC(C(=O)NCCNC(=O)CN2CCOCC2=O)CC1=O c1(N(C)CCC2CC2)ccc(S(=O)(=O)NCC(O)CCC2CC2)c(Br)c1 C=C(CNC(=O)C(c1ccccc1)OC(C)C)CCNC(=O)CC1CSCCS1 c1(CC)ccc(Cl)cc1.C12(C)C=CCN1C(=O)N2C1CC(C)N(C(=O)C(O)O)C1 C=CC(C)(CCOC)C(=O)NC(C)CCCNC(=O)CC1CCCNC(=O)C1 C1(CCN(C2CCOCC2)CC#C)CN(C(=O)OC(C)(C)C)C(C)(C)CO1 N1(C(C2C(=C)C2)=O)CCCCC1CCN(C(=O)C(CC)=CC)C C=Cn1nccc1C(=O)NC1CC(CNC(c2ccc(C(C)(F)F)nc2)=O)C1 c1(COc2c(OC)ccnc2SC)ccc(F)c(Cl)c1F C(=O)(CCCN=[N+]=[N-])NC(C=CC(=O)Nc1c(C)n(C)nc1)C C1(C(N2CCC(N(C(c3ccc(F)s3)=O)CC)C2)=O)CCCC(OC)C1 N1(S(CC)(=O)=O)CCC(C(N2CC(C)(NC(C3CCOC3C(=O)O)=O)C2)=O)CC1 CCC(CC)CC(=O)NCCN(CCCN(C)C)C(=O)CC1CCC1S(C)(=O)=O c1(-c2nn[nH]n2)ccc2c(c1)C(=O)N2.C1(COCCOC)CCC(C)S1 CCC(C(=O)NC(C1CCN(C(c2cncc(C3CC3)c2)=O)C1)(C)C)C(C)C C1(C(N2CCC(C3CCCCN3C(=O)C=Cc3ccco3)C2)=O)C2CCCCC12 C(=O)(CCCCCSC)NCC1C=CC(NC(c2n(CC)nc(C(C)C)c2)=O)C1 CC(C)C(C)(CN=c1[nH]c(=NCCC(C)CO)[nH]c2cc[nH]c12)N1CCOCC1 CC1(C)CCN(C(=O)C=C2CCC2)CC1C(N1CCCSCC1C)=O c1(OC)cccc(C(C2C3CCC2CC3)NC(C2(c3ccccc3)CC(F)C2)=O)c1 c1(C(N2CCC(CN(C(C(C(CC)CC)C)=O)C)C2)=O)cc2c(cc1Cl)OCO2 c1(OC)ccc2c(c1)CN(N1C=C3C(=O)N(C(C)(C)C)C=C3C1=O)CC2 O(NC(=O)CCCC(CC)NC(C1(C)CNC(=O)N1)=O)CC#C C1(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)CCCCC(C)(C)C1 N1(C(c2ccc(O)nc2)=O)CC(C2CN(C(c3cnc4n3CCS4)=O)C2)C1 CC(CC(=O)N(CCCCN(C(=O)CN1CC2C=CC1C2)C)C)CC(C)(C)C c1(C(N(CCOCCNC(C(C)CF)=O)C)=O)cc(F)c(O)c(F)c1 c1(C(N2CCC(CS(=O)(=O)C3CC3)CC2)=O)n[nH]c(=O)c2ccc(Br)cc12 c1(C(=O)NCCCCCNC(CCOCCOC)=O)ccc(C)c(P(C)(C)=O)c1 c1(CC)cc(C(N2CCC(C)(NC(=O)CC(C)SC)C2)=O)cc(N)c1 C1(NC(C(=O)N(C)Cc2ccc(C)cc2)=O)CC(O)CN(C(=O)OC(C)(C)C)C1 CC(C)CC(C)(C)C(=O)NCC1CCC(C(N2CCCCCC2C)=O)O1 O(NC(=O)CC=Cc1ccccc1)CC(=O)NCc1c(CC)nn[nH]1 C12(C3CCCO3)CC1CN(C(c1cnn(CC(F)F)c1)=O)C2.C(C)(CC(=O)N)SC Cc1cc2ccc(C(=O)NC(CNC(=O)CC3(C)CCCCC3)C3CC3)cn2c1 C1(NC(CSCc2nc(C)sc2)=O)CC2CC(NC(=O)Cn3cnnc3O)C1C2 N12CC3CCN(CC13)N1CCCC(C1)C2=O.C(=O)(CCS(C)(=O)=O)OC C1(=CC(=O)NC(C2CCN(C(=O)Cc3csc(Cl)n3)C2)(C)C)CCCCC1 C1(O)(C(CNC(c2c(C)noc2)=O)C)CCN(C(=O)C=CBr)C1 N1(C(c2c(C)ccn2C)=O)CCC(C2(NC(=O)CN3CCCNC3=O)CC2)C1 c1(C(N2CC3CC2CN3Cc2cccc3cncn23)=O)ccc2ncsc2c1 N1(C(c2cc(C(=O)OC)cc(F)c2)=O)CCC2(CC1)CC2n1ccnn1 C(CCCCC(=O)N1CCCN(C(C2CCCCC2C(F)(F)F)=O)CC1)OC c1(C(=O)NC2CCCCN(C(C(C=C)C)=O)C2)cc(C)cc([N+](=O)[O-])c1 c1(NC(COC)=O)cccc(C(=O)NC(c2ccc(CC(F)(F)F)cc2)C)c1O c1(OC)ccc2c(c1)CCC2C(=O)Nc1ccccc1-n1cccn1 C1(CC(=O)N(CC(CN(C(C)=O)C)O)C)CC(O)CN1C(=O)CN1CC=CC1 N(C1CCc2c(C(F)(F)F)cccc21)C(=O)CC1CCCC(C(F)(F)F)N1 c1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2CCO)=O)nccn2nccc12 C1(C(=O)NCCCCCCNC(CC2C(CC)C2)=O)CC(=O)c2ccccc2C1 C1(CNC(C=CC(C)(C)NC(c2c(C)nccn2)=O)=O)C(=O)NCCC1C C(=O)(C1=C(Cl)CC1)N1C(C(CNC(C(CC)O)=O)(C)C)CCC1 N1(C(C=C(C)Cl)=O)CCC2CCC(C1)N2C(=O)Cc1ccc(O)cc1Cl N1(C(N)=O)CCCC(C(N2CC(O)(CNC(C34CC(CCO3)C4)=O)C2)=O)C1.C(=O)(C1CC1)N CC1CN(C(c2cncc(CO)c2)=O)CC(C)CN1C(=O)C(CO)C(C)(C)C N1(C(Cc2cnc(C)s2)=O)C2CCC(C(N3CCCCC(CO)C3)=O)C1CC2 Cc1nc(=N)[nH]c(=NCC2CCCC2NC(c2ccnn2CC(C)C)=O)[nH]1 N1(C(C2CCCN(C(CC)C)C2)=O)CCOC2(C1)CN(C(=O)OC(C)(C)C)C2 C1(N(C)C)CCCN(C(=O)CONC(C2CCOC2(C)C)=O)C1 C1(OC)CC(C)CN(C(C2CCCN(C(=O)CC3CCC(=O)C3)C2)=O)C1 N1(C(c2cc(C)sc2C)=O)CCC(C)C(CNC(c2nccc(C)c2N)=O)C1 CC1(C(=O)NCc2ccc(C(=O)N(C3CC3)CC3CC3)cn2)CCC(O)CC1 C1(C(N2C(CC(N3CC=C(C)CC3)=O)CC2)=O)CC12CCCCC2 Cc1nn(C2CC2)cc1C(=O)NCC1C2CN(C(C34CC5CC3C4C5)=O)CC12 c1(N)cccnc1.n1(CC(=O)N(C)C)ccnn1.C12(CC1)C(=O)NCCC2 C(N=c1[nH]c(=NCCF)[nH]c2ccccc12)c1n(C)ncc1Cl Cc1ncsc1C=CC(N1CCC(NC(C2CCCCS2)=O)CC1)=O O(N(C)C(=O)CCN(CC(C)C)C(c1cc(Cl)cn1C)=O)CC(=O)OC N1(C(Cn2ncc(CC)c2)=O)CCC(F)(CC(N2CCCC3(C2)N=N3)=O)CC1 CN1CC=C(CC(=O)N(C2(CC(N3CCC4NCCC4C3)=O)CC2)C)CC1 c1(C(N(C2CCCN(C(COCCC=C)=O)CC2)C)=O)cnn2c(=N)[nH]cnc12 N1(C(C2C(COC)C2)=O)CCN(C(C2OCCO2)=O)CC1c1ccccc1OC C1(CNC(C2CCS(=O)(=O)N2)=O)CC2(CCC2)CN1C(c1cn2ccsc2n1)=O N1(C(COC(C)=O)=O)CC2(C1)CN(C(C1CN(S(C)(=O)=O)C1)=O)CCO2 C1(NC(c2on(C)c(=O)c2)=O)CN(C(=O)CC2=CCCC2)CC2(CC2)C1 C=CC(C)(C)CC(=O)NC1CCN(C(c2ccc(SCC)nc2)=O)C1(C)C N1(C(C=C(CC)CC)=O)CCc2[nH]nc(CNC(c3ccncc3Br)=O)c2C1 c1(C(N2CCCC(NC(CCCCCC)=O)C(F)C2)=O)cc([N+](=O)[O-])ccc1N Cc1cc(CC(=O)NC(C)(CNC(c2c(C)n[nH]c2C)=O)C(C)C)n(C)n1 n1(CC(=O)NC(CNC(c2cocc2Br)=O)C2CC2)cc(C2CC2)cn1 c1(C(=O)NCC(C)NC(c2cc3cc(F)ccc3[nH]2)=O)n[nH]c2c1CN(C)CC2 CCCC(C)C(=O)N1CCC(CC(=O)Nc2ccccc2CC(N)=O)C1 c1(C(=O)NC2CCCN(C(c3[nH]c(=NC)sc3)=O)CC2)ccc2nccnc2c1 C1(CC=C)(C(=O)N2C(C)CC2)CCCC1.c1(C(=O)NC(C)CC)ncn(C)n1 C1(C(=O)NCc2c(C(=O)NC(C)COC3CC3)n(C)nn2)CC12CCOCC2 N1(C(CC(=O)OCC)=O)CC(CNC(=O)C(C)Cc2ccccn2)OC(C)(C)C1 Cn1nnc(C(=O)NC2CCN(C(C3CC(O)(c4ccccc4)C3)=O)C2)n1 c1(C(N2C(CNC(c3c(C)csc3Cl)=O)CCC(C)C2)=O)ccc2nncn2c1 C1(O)(C(=O)NCC2C(NC(c3cnc(C(C)O)s3)=O)CCC2)CCCC(C)(C)C1 CC1(CNC(=O)CC2(NC(c3ccncc3F)=O)CCC2)CCC(=O)N1 c1(C(=O)NC2(C)CC(NC(COC(CC)C)=O)C2)cccc(C)n1 N1(C(CC2CC(=C)C2)=O)CC(F)(F)C1C1CC1ONC(CC(O)C(C)C)=O c1(OC)ncc(Cl)c(=NCC2CCCC(NC(C3CN(C(C)=O)C3)=O)C2)[nH]1 C(=O)(CCCC(F)(F)C(F)(F)F)NCCN(C(c1occ(C)c1)=O)C CCC(C)(C)CC(=O)NCCC1(C(=O)N(CCS(N)(=O)=O)C)CCC1 CC1(NC(c2ccnnc2)=O)CCCN(C(=O)CC2CCC23CCC3)C1 C(CCC(C)C)(C(=O)NCC(c1cn(C)cn1)O)NC(CN(CCC)C)=O C(N=c1nc2c(cnn2C)c(N2CCC(C(C)C)CC2)[nH]1)c1cccc(SC)c1 N1(C(c2n(C)ncc2C2CC2)=O)CCC2CN(C(=O)CC3CCCOC3)CC2C1 n1(C(C)C(=O)NCCC2CC2(Cl)Cl)cc(C2(C)CCCO2)nn1 N1(C(C2CC(CC)(CC)C2)=O)CCCCC1CC(=O)NC(CC)C(F)(F)F CCCC(C(=O)N1CCCC(CCNC(C2(CO)CCOCC2)=O)C1)S(N)(=O)=O N1(C(C(CC(=C)C)C)=O)CCCCC(C2CN(C(=O)Cc3cn(C)nc3C)C2)C1 c1(C(N2CC3CC2C3NC(C2(CO)CCOC2)=O)=O)cnc2c(n1)CCCC2 N1(C(Cc2ccc(C)cc2)=O)CCC2(CC2)CC1C(N1CCCCC(CO)C1)=O C1(NC(COc2cccc(C)c2)=O)CC2(CCN(C(c3ccc(Cl)s3)=O)CC2)C1 N1(C(CC)=O)CCN(C)CC1CNC(c1sc(C2CC2)nc1C)=O c1(C(=O)NC(C(C)Nc2ccncn2)(C)C)ccc(C2CC2)cc1F C1(NC(C(C2CN(C(=O)CCC3CCCC3)C2)OC)=O)CC12CCCCCC2 CC1=C(C(=O)N2CCC(CC(=O)NCCNC(=O)C3CC3)CC2)CCC1 c1(CC)ccc(OC)cc1.O1NC(=O)CN(C)C(=O)C1 C12(C)CC(NC(=O)C(O)C(C)SC)(CN1C(=O)C1=C(C)OCC1)C2.CO N1(C(CN2C(C)CCC2)=O)CCC(C(=O)Nc2cccc(O)c2)(CO)C1 C=CCN(OC)C(=O)c1cn(CCNCC)nn1.C1(=O)C(CCC)O1.OCC C(CCC(C(=O)NC(COC)CO)NC(C1CCC2(CC1)CC2)=O)OC c1(C(N2CC(Cn3cc(-c4cccc(C)c4)nn3)C2)=O)cc2c(C)sc(C)c2s1 C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CC(NC(c3cc(C)c(C#N)cn3)=O)C2)C1 C1(NC(C2C(C)OCC2)=O)CN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(=O)OC(C)(C)C)CCC=CC1C(=O)OCC1CC2(C1)CC2F C1(CC)CC(C(=O)NOCC2(C)CC2)CCN1C(=O)CCc1cccn1C N1(C(COCc2n(C)ccn2)=O)CCCOC(CNC(C23CCC(C2)C3)=O)C1 Cc1cc(C(=O)NC2CC(C)CN(C(=O)C(C)NC=O)C2)cc(O)n1 C1(C(C)(C)C(=O)NC2CC2F)CCCN(CCO)C1.C12CC(C1)NC2=O C=CCN=c1[nH]cc(C(N2CCC(NC(C3(CCF)CCC3)=O)C(C)(C)C2)=O)s1 CC1=C(C(=O)NC2CCC(NC(c3cncc(C(F)F)c3)=O)C2)CCO1 C(=O)(C1=CCC2(COC2)OC1)NC(C(C)NC(=O)Cn1ccc(C(F)F)n1)C N1(C(C(CCSC)NC(N)=O)=O)CCC(NC(c2sccc2C)=O)CC1C N1(C(CCOCCOC)=O)CCC(C(N2CCN(CC(=O)N(C)C)CC2)=O)C(O)C1 CC1CN(C(c2ccc3c(c2)COC3)=O)CCCN1C(=O)Cn1cnc(=N)[nH]1 c1(OC)c(F)ccc(C(N2CC3CN(c4cc(C(C)C)ncn4)CC3C2)=O)c1F N1(c2n(C)c(=O)n(C)c(=O)c2)CCC2CCC(C1)N2C(=O)CC1CCC2CC2C1 c12cc(ccc1Cl)NC(=O)C(=O)N2.C1(CC(=O)OC)CCC(c2ccccc2)C1 C1(CC)C(=O)NCCCN1C(=O)CCN(C(c1cc(C)c[nH]1)=O)C1CC1 Cc1ccc2c(c1)CCC(C(N1CCC(CNC(C34CCC(CC3)C4)=O)C1)=O)O2 C(=O)(CC(C(=O)NCCC(C)CCNC(c1cnsc1)=O)NC(C)=O)OC c1(CCC)ccc(C(=O)NC2CCC2CNC(=O)C(C)(C)n2cc(Cl)cn2)s1 C(c1ccc(F)cc1)=CCC(N1CC2C(CNC(CCSC)=O)C2C1)=O N1(C(c2c(N)cc(F)cc2)=O)CCC(C2CC2)C1CNC(=O)CN1CC=CC1 CC1CSCC1NC(=O)C(=O)NC(C1(c2ccccc2)CC1(C)C)C1CC1 C(N=c1cc[nH]cc1S(=O)(=O)NC(C)CC1CCCO1)c1c(C)occ1 N1(C(CC(c2c(C)n[nH]c2C)CO)=O)CCCN(C(=O)Oc2ccccc2)CC1 c1(OC)ccncc1C(N1CCCC1CNC(c1nccnc1N)=O)=O CC(O)C(C)(C)C(=O)Oc1cccc(C(=O)NC2(n3cncn3)CC2)c1 CCCC(CC(=O)NCC)N.c1(CN(C(=O)OC(C)(C)C)CC)cccc(F)c1C c1(C(N(C2CC(C#N)C2)CC(=O)NC(c2ncc[nH]2)CC)=O)ccc(Cl)o1 C1(NC(c2cn3c(n2)COCC3)=O)CCC2CN(C(C34CC3C4)=O)CC2C1 c1(C(=O)NCCCCNC(CSCC=C)=O)coc2c(C)cccc12 C1(CNC(CCCCSC)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 N1CCC2(CC(C(=O)N=c3[nH]ccn4ccc(Br)c34)C2)C1.O=CC1CCc2scnc21 N1(C(C=CCOC)=O)CCC(C(N2CC=CC(OC)C2)=O)(CO)C1 C(=O)(C1CCN(C)c2ccccc21)N1CC(C)N(c2ccncc2[N+](=O)[O-])CC1 O=C1CN(CC(=O)NC2CCCCC2NC(C2CC3CCC2C3)=O)C(=O)N1 C1(c2cn(C(CC)C)nn2)CN(C(=O)CC(C)C2CCCO2)CCO1 C(=O)(C(C)(C)N(C)C)NC(C1(O)CN(C(=O)CCCc2ccsc2)C1)C C(=O)(CCC(C)NC(c1ncn(C)n1)=O)NCc1ncc(C)o1 C=CCC(CNC(=O)CC1(N(C)C(c2cncc(O)c2)=O)CC1)CC(C)C C1(NC(C23CC(F)(C2)C3)=O)CN(C(c2csc(-c3nc[nH]n3)n2)=O)CC12CC2 N1(C(c2n(CC)nnc2C)=O)CCCC2(CCCN2C(C23CCC(C2)C3)=O)C1 C1(C(=O)NCC2CCN2C(c2n[nH]cc2Cl)=O)(COC)CCCO1 CC1CC(=O)NC(C(N2CC3C(CNC(=O)C=C4CCOCC4)C3C2)=O)C1 C1(NC(C2(C)CCOC2)=O)CCC(NC(=O)CNC(=O)C2CC2)CC1 C1(C)(C(=O)NCC(n2cc(C(C(C)C)O)nn2)C)CC(F)(F)C1 c1(C(N2CC3CN(C(CC(C)CN(C)C)=O)CC3C2)=O)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=C(C)CC2)=O)C2CCC1C(NC(c1cc(C)n(CCO)n1)=O)C2 c1(CC(N2CC3(CN(C(=O)CCc4cnn[nH]4)C3)C2)=O)cncc2ccccc12 C1(CNC(c2c(C)nc[nH]2)=O)CC2CCC1N(C(c1cc(C3CC3)nn1C)=O)C2 c1(C(=O)NC2CC3(C2)CN(C(=O)C=C2CCC2)C3)cccn2ncnc12 C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCC1NC(C12CC3CC1C2C3)=O N1(C(C(CC=C)C)=O)CCC(CNC(=O)CCOCC(C)(C)C)CC1C N1(C(c2ccn(CCCC)n2)=O)CCC(NC(C2CCCC3(CC3)C2)=O)C(O)C1 c1(C(N(C)CC2CCN(C(c3c(C)nc(CC)o3)=O)C2)=O)cc(F)cc(F)c1N O=C(C#CC1CCCCO1)N1CCC(F)CC1F CCCC(C(=O)N(CC(O)CNC(c1ccn(CCN(C)C)n1)=O)C)C(C)C N1(C(CN(CC)CC)=O)CC(C(=O)NC(C2CCCO2)CO)C(C(C)C)C1 C1(NC(C(C)=C(CC)C)=O)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1C C(CCC)(C(O)C(=O)NC(C)C(=O)NCC(C)C)NC(C(COCC)C)=O C1(N(C)CC2(O)CCC2)CCCN(C(=O)CCN2CCOCC2)C1 N1(C(C2(N(C(=O)CC3COCCN3C)C)CC2)=O)CC2C(CN)C2C1.CCO N1(C(C(C)NC(CC)(C)C)=O)CC(NC(=O)Cc2ccn(C)c2)CC1(C)C C12(NC(CCNC(=O)OC)=O)CC(C(=O)NCCCc3cc[nH]n3)(C1)C2 C(CN=c1[nH]c(=NCCc2nc(C(C)(C)C)cs2)[nH]c2ccsc12)NC(=O)OC N1(C(=O)C(=O)NCC2(CF)CCC2)CCC(c2cccnc2)C1 c1(C(=O)NCC2(F)CC(NC(C3C(C(N)=O)CCC3)=O)C2)c[nH]ccc1=O C1(N(C)C(c2cscc2F)=O)CCCC(NC(=O)Cn2nnnc2C2CC2)C1 c1(NCCNC(=O)C2CC2)ncc(C#N)cc1Cl.c12ccccc1N2 Cc1ccc(C=CC(=O)NCC(C)CNC(c2c(Br)cnn2C)=O)s1 C1(C)(CC)CCC(C(=O)NC2CC2CNC(=O)CCc2cn[nH]c2)O1 c1(OC)ccc(Br)c2c1C(NCC1CCN(c3ccc(F)cc3)C1=O)CC2 C(=O)(C(C)CS(C)=O)N1CCN(C(c2nnc(C)s2)C)CC1.c1(CC=O)ccccc1 Cc1ccc(C(=O)NC(CNC(=O)Cn2cc(C)cn2)C(C)C(C)C)c(O)c1 CC(C)(O)C(C(=O)NCCn1cccn1)NC(=O)C(F)CC1CCC1 c1(C(N2CC(C)=C(CNC(C(C)(C)NC(C)=O)=O)C2)=O)cc(F)cc2cnccc12 O(NC(=O)C(CCC(C)C)NC(=O)C(C)NC(N)=O)C(CC)CC c1(OC)ccc(CCC(=O)NCC2C(C)CCCN2C(=O)CSC(C)C)cc1C C=CCC(C(=O)Nc1cccc(C(=O)NCCn2cnc(C)c2C)c1)OC C=CC1(C(=O)NC(c2c[nH]ccc2=O)C)CCN(C(=O)CC(C)C(F)F)C1 N1(C(C(C2CC2)OC)=O)CCN(C(c2ccsc2)=O)C(C2CCCC2)C1 N1(C(C(=O)N(C)C)=O)CCC(NC(=O)Cc2ccn(C(F)F)n2)C(F)C1 Cc1cc(=NC(=O)CN2CCC(F)(F)C(CNC(=O)CC3CC3(C)C)C2)[nH]o1 C(CCO)(C(C)(C)C)NC(C=CCN(C)C(c1cnc[nH]c1=N)=O)=O N1(C(C(C)(C)CO)=O)CC2CN(C(C3(S(C)(=O)=O)CCCC3)=O)CC2(C)C1 CC1CN(C(c2cnc(C3CC3)nc2)C(=O)NCCC#N)CC1(C)CO c1(C(N2CCCC(N(C(C3CC(C)N(C)C3)=O)C)C2)=O)c2c(nn1C)CCOC2 N1(C(C(COCC)N=[N+]=[N-])=O)CCCC(C2CN(C(c3cc(=O)cc[nH]3)=O)C2)C1 Cc1nc2c(s1)CCCC2C(=O)NC(C)CNC(c1coc2ccc(O)cc12)=O c1(C(N(C(CCNC(C(C)OCCCC)=O)C)C)=O)cc(C)n(C)n1 n12cc(nn1)NC(=O)NCC1CC21.N1(C(C)(C)C)CCOCC1.C1(CNC)CN(C=O)C1 C1(C(=O)OC)CC12CCN(C(c1cc(F)c(-c3cnn(CCO)c3)cc1F)=O)CC2 CCCC(CCC)C(=O)N(CCNC(C1CCCC1C1CC1)=O)CCOC c1(COC(c2cn(Cc3ccc(C)cc3)nc2)=O)cc(O)n2nccc2n1 C#Cc1ccc(F)c(C(N2CCCN(C(c3ccsc3OC)=O)C(CO)C2)=O)c1 c1(C(N2CC(O)(CCNC(=O)CCCF)C2)=O)ccc(N2CCC(O)CC2)cc1 C1(C(=O)NCCCC(CO)NC(C=C2CCN(C)C2)=O)CCOC(=O)CC1 C=C(F)C1(CC(=O)NC2CCOCC2C(=O)NC2CC(CC)C2)CCC1 C12(CNC(=O)C(O)Cc3ccccc3)CC1CN(C(=O)CC1(CO)CC1)C2 c1(NC)c(C(N2CCC(NC(C3(OC)CC3)=O)C(CO)C2)=O)cccc1[N+](=O)[O-] C1(NC(CC(C)OC)=O)CCCN(C(=O)C(c2ccccc2OC)C)C1C C(C)(C(=O)NC1CCOC(C(=O)NC2CC(O)C2O)C1)(C(C)C)OC C#CCCCCCCC(=O)N1CC2CC1(C(=O)NCCC(=O)OC)C2 Cc1ccc(C(N2CC(NC(=O)Cc3cc(C)[nH]n3)CC(C)C2)=O)cc1CO c1(CC)cnc(O)c(C(=O)NC2CCN(C(c3ccc(O)cc3)=O)CC2CO)c1 c1(C(N2CCN(CC3(NC(C(C)SC)=O)CC3)CC2)=O)cc(F)c(F)cc1F N1(C(c2c(CC)ccc(F)c2)=O)CCC2(NC(=O)Cc3cccnc3)CCCC12 C12(CC3(CC3)C1)C(=O)OC2.C1(C(CC)C)CN(C(C2CC2C(=O)N)=O)C1.C1(O)CC1 C1(C(=O)NC(CCNC(C2CCC(CCCCC)CC2)=O)C)CC(C)CC(=O)N1 c1(CN2CCCCC(NC(CN(C)C)=O)C2)cc([N+](=O)[O-])c(Br)cc1F C1(N(C(c2c(CC)scc2)=O)C)CN(C(=O)CSc2nncn2C)CCC1O C1(C(=O)N(CCc2ccccc2)Cc2cnn[nH]2)CC12CCN(CCCO)CC2 Cc1nc(C(C)C)nc(O)c1C(=O)NCCC1CN(C(=O)C(C)C2CCCC2)C1 CN1CC(C(=O)NC2(CNC(c3cc(C(N)=O)c[nH]3)=O)CC(F)(F)C2)NC1=O c1(C(N(C)CC2(NC(C(CC=CC)C)=O)CC2)=O)cc(Br)c(C)cc1F C(CCCC(=O)NC(C(=O)N(C)Cc1cnc[nH]1)c1cccs1)SC c1(C(=O)NC2C3CN(C(c4c(N(C)C)ccnc4)=O)CC32)ccc(F)c(F)c1F C12(C(=O)NC(C(C)F)C)CCCC1CCN2C(=O)C(c1cnn(C)c1)C C1(NC(c2c(C(C)C)cccc2)=O)CN(C(C2(C3CC3)CC2)=O)CC2(CCC2)C1 C=CC(CC)C(=O)N(C(C(=O)NC(C1(OC)CCC1)C)C1CC1)C N1(C(CCc2onc(CSC)n2)=O)CCC2(NC(=O)Cc3cnn(C)n3)CCCC12 N1(CC)CC(NC(=O)C(CC2CC2)NC(=O)C=Cc2cncs2)CC1=O c1(C(C(=O)NC(C2(O)CN(C(C3(O)CC(C)(C)C3)=O)C2)C)CO)ccc(F)cc1 C1(NC(C(C)C2CC2)=O)CCC(N(C)C(c2cccc(Cl)c2)=O)CC1 c1(CC)ccc(C)c(NC(=O)CC(c2ccnn2C)NC(C2CC(C3CC3)C2)=O)c1 C1(C(N(CC(C)NC(c2c(C(=O)OC)n(C)nc2)=O)C)=O)CN2CCC1(C)CC2 N1(C(C(CCC)O)=O)CC2CCC2(CNC(=O)CN2CC(=O)N(C)C2=O)C1 c1(CC(C(=O)NCC(CNC(CC(=C)C)=O)C)O)ccccc1Cl Cn1cc2c(n1)CC(C(=O)OCC1CN(S(C)(=O)=O)CCO1)CC2 Cc1coc(C(=O)NC2CCC(CCNC(=O)C(F)(F)c3sccc3C)C2)c1 N1(C(CC(=O)OC)=O)CCC(NC(c2nc(Cl)sc2C(C)C)=O)C(CO)CC1 C=C(C)CCCC(=O)NCCC1CN(C(=O)COc2ccccc2Cl)CCO1 C1(Cc2ccccc2)CNC(C2CCC2)CO1 Cc1cc2cc(C(=O)NCC3OC4CC3C4)ccc2cn1 C1(CC(=O)N(C2C(N(C)C)COC2)C)CCOC1(C)C S(=O)(=O)(c1ccsc1C(N1CCC(NC(=O)C=Cc2cncs2)C(O)C1)=O)NC Cc1ccccc1C(=O)NCC(=O)NCC(F)CNC(c1sccc1Cl)=O CC1(C)OC2(C(=O)NCCCCNC(C34CCCC3C4)=O)CCC1CC2 c12c(C)ccc(C)c1NC2=O.n1(CCOC)cc(Cn2ccc(C(=O)O)c2)nn1 N1(C(C=C(C)Cl)=O)CCC2CC(NC(c3cnc4nccn4c3)=O)CCC2C1 c1(C(N2CC(O)(CNC(c3ccc(SC)o3)=O)C2)=O)cnc2c(c1)CNC(=O)N2 S(=O)(=O)(c1ccc(F)c(Br)c1)N1CCN(C2CCN(C(=O)C(F)F)C2)CC1 C1(NC(CCC2N(C(C=CC(CC)C)=O)CCC2)=O)COC2(CCCC2)C1 N1(C(C(C)OCC=C)=O)C(C(=O)NC2(C(N)=O)CC2)C2CC(O)C1C2 C1(CC)C(C(=O)NCCCC(C)(C)OC)CCN1C(c1cc(C(N)=O)c[nH]1)=O c1(CN(c2nnc(Br)s2)C)ccc(Cl)c(C2=CCNCC2)n1 c1(C(N2C(C(C)NC(c3cnc(O)o3)=O)CCCC2)=O)cccc2oc(O)nc12 N1(C(C(CC)COC)=O)CCCC(NC(c2ccc(Cl)c(Cl)c2)=O)C1C N1(C(c2c(C)cccn2)=O)CC2CCC(CNC(C3(F)CCOC3)=O)C2C1 C1(C(=O)NC(CCCCNC(=O)Cc2ccns2)CO)CC2CCCC(C1)C2 c1(CNC(c2c(NC(=O)OC(C)(C)C)nccn2)=O)ccnc2c1CCO2 Cc1[nH]nc2cc(C(=O)NC(C)(C)CC3CCC3)ccc12 c1(C(N2CCCC(N(C)C(C3CC4CC3C4)=O)CC2)=O)c[nH]c2cc(O)ccc12 C1(NC(c2ccsn2)=O)CC(NC(c2ccnc(O)c2Br)=O)C12CCC2 CCC(CC(C)C)C(=O)NC(CN(C)C(c1sc2ccsc2c1C)=O)CC C1(NC(C2CCN(C(C)C)CC2)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)C1(C)C C1(S(=O)(=O)NC)(C(=O)OC(C2CNCCO2)C(=O)OCC)CCC1 c1(N2CCC(NC(C3C(=C)CC3)=O)C2)cccc(Cl)c1Cl C12(C(=O)NCCCOC3CCN(C(C4CC5CC5C4)=O)CC3)CCOC1CCOC2 Cc1nn(CC(=O)NC(C(C)NC(C2(O)CCC2)=O)C(C)C)c(C)c1[N+](=O)[O-] CC(C)(C)C(CNC(=O)CCC(F)(F)F)C(=O)NC1CCC2CCC12 c1(NC(c2cccc3nccn23)=O)cccc2ccoc12 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CCC(C)C)CCC12CCC2 CCCCCS(=O)(=O)CC(=O)N(CC(C)CNC(=O)CC12CC(C1)C2)C C(C(F)(C(=O)NC(C)C(=O)NCCF)C(C)C)NC(c1c(CC)cccc1)=O CC(C)C(C(=O)NC(C)CN(C)C(c1n[nH]c(=N)s1)=O)c1ccncc1 c1(OC)ccc(NC2CCC(C)(CNC(=O)OC(C)(C)C)C2)cc1N1CCOCC1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(C2CN(C(c3c[nH]c(=N)o3)=O)C2)C1 CN1C2CCC1CN(C(=O)C(CO)NC(c1ccncc1N)=O)CC2 Cc1cc(C(=O)NCCNC(C2(Cc3ccncc3)CCC2)=O)cc(C(F)F)c1 c1(OC)cnncc1C(=O)NC(C1CCN(C(C2CCC(=O)N2)=O)C1)(C)C CC1CCC(NC(c2cnc(-c3ccccc3)[nH]2)=O)CN1C(=O)CNS(N)(=O)=O c1(C(N2CC(C)N(C(=O)CN3CCCC3=O)CC2)=O)c(F)ccc(N)c1F CCCC(C)CC(C(=O)Nc1ccc(Cl)cc1)N1CCN(CC2CCOC2)CC1 C(=O)(CCCCCF)N1CCC(C(C)NC(CCc2cccc(OCC)n2)=O)C1 C(CCC(C(=O)NCC(C)C)N1CCOC(C2CCCOC2)C1)OCC=C C(CN(C)C)(C(=O)NCC(C)(O)CO)NC(CNC(=O)OC)=O CCCC(CC(C)C)C(=O)NC(CNC(C12CC(C)(C1)OC2C)=O)C1CC1 N1(C(C(C)=C(CC)C)=O)CCC2CCN(C(=O)Cc3ccn(C(F)F)n3)CC2C1 C(CCCCCCO)NC(C(C1CCCN(C(=O)C=CC(=O)N(C)C)C1)C)=O Cc1cc(C(=O)NCCC(C)N(C(=O)Cc2ccc(Cl)cn2)C)ccc1C#N N1(C(C2(C)CCCO2)=O)CCC2CCN(C(c3nc(Br)cnc3N)=O)C2C1 c1(NC(C(C)C)CCN(C)C(c2ccsc2)=O)ccc(C#N)cc1[N+](=O)[O-] Cc1cccc(C(=O)NC2(CCNC(=O)C(F)C(C)(C)O)CCCC2)c1C CN1CCN(C(c2cnc(S)n2C)=O)CC1CNC(=O)CCN1CCCCC1 c1(CC(=O)NC(CN(CC)CC)C)cscc1Br.C12(CCC1)C(=O)OCC2 C(=O)(C(C)(C)n1cc(Cl)cn1)N(CCCNC(C(C1CCCOC1)OCC)=O)C N1(C(c2n(CC#C)cnn2)=O)CCN(C(c2scnc2Cl)=O)C(CC)C1 C1(C(=O)OC)CC(C(=O)OC)CC(C(N2CCC(C(C)N)CC2)=O)C1 Cc1cc(C(=O)NCC2CCCC(CNC(C3(N4CCCC4)CC3)=O)C2)n(C)n1 C#Cc1ccnc(C(N2CC(N(C)C(c3nc(CSC)no3)=O)C(C)(C)C2)=O)c1 C(CC(C)C)(C(=O)NC1COC(C(C)C)C1)ONC(c1c(CC)n(C)cc1)=O c1(N(C(=O)CCSc2ccccc2[N+](=O)[O-])C)cc(Cl)cc2c1OCC2 CN1C(=O)CCc2ccccc2CC1=NCC1(O)CN(C2CCOCC2)C1 CCC(O)C(C)C(=O)N1CCC(C(C)(C)NC(=O)Cc2cnn(CC)c2)C1 C(C1CCCCCC1)=CC(=O)NCC(=O)NCC1CCCCS1(=O)=O C1(NC(c2cncc(CNC(=O)Cc3cnccn3)c2)=O)CCCCC1(F)F C1(CNC(c2cccs2)=O)CC2(CO1)CN(C(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 c1(OC)ccc(C=CC(=O)NC2(CCNC(=O)Cc3ccns3)CCC2)cc1O C1(CNC(COCCCCC)=O)COC(C)(C)CN1C(c1cccc(C)c1)=O C12CN(CCC1C)C(=O)C2.C1(CCC)(CC)CCCN1C(=O)CCC1CC1 Cc1ccc(N2CCC(CC3CN(C(=O)NC4C(C)(C)C4(F)F)CCO3)C2)nc1 C1(NC(Cc2c(C)n[nH]c2C)=O)CC2CC(C1)N(C(=O)Cc1cncnc1)C2 c1(C(=O)NC(c2nn[nH]n2)C)ccccc1OCCCC#N CC(C)C(CNC(=O)C(C)n1ccnc1)C(=O)NCCCOC(F)(F)F C=CC(CC)CC(=O)N1CCCC(CNC(c2coc(-c3cn[nH]c3)c2)=O)C1 C1(C)(C(=O)NCC2N(c3ncc(OC(C)C)cn3)CCC2C)CCCCCC1 c1(NC(=O)CN2CCN(C(=O)NCc3ccncc3)CC2)cc2cccnc2o1 c1(C(N2C(CN(C(=O)C(N)=O)C)COCC2)=O)cc(=O)c2ccc(Cl)cc2o1 N1(C(c2cncc(OCC)c2)=O)CCNc2ncccc21 c1(OCCC)cccc(C(=O)NCCC2CCN(C(=O)C(C)c3ccsc3)C2)c1 C1(C(=O)NCCCN(C(CCOC)=O)CCO)CC2(C)CCC1(C)O2 C1(CC(=O)NCC2(OCC)CC2)C2CN(C(C3CCN(C)C3=O)=O)CC12 N1(C(CCOC(Cc2ccc(C)cc2Br)=O)=O)CCCC2CCCCC12 N1(C(Cc2ccc(S(C)=O)cc2)=O)CCC2(CC1)CC(NC(C1CC1(C)C)=O)C2 c1(CNC(C(c2cc(OC)c(F)cc2)(C)C)=O)cc2c(F)c(F)cc(F)c2[nH]1 c1(C2C(COC)C2)ccc(NCCC2(NC(=O)C=CCF)CCC2)nc1 CC(O)(C(=O)N1CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(F)C1)C(F)(F)F C(=O)(C1=CCc2ccccc21)NCCC(CCNC(CC(=O)OCC)=O)C c1(CC(=O)NC2CC(C(C)NC(=O)CCC3CCCOC3)C2)cc(C)nn1C c1(C(=O)NCC2(F)CCN(C(c3ncc(OC)nc3)=O)C2)ccc2c(c1)CCC2 c1(CC(N2CCC(NC(COCC(=O)NC)=O)C2C(C)C)=O)cccc(C)c1C C1(C2(C)CC2)CC(O)CN1C(C1CCCN1C(C1CCC(F)(F)C1)=O)=O C(=O)(C(C)(C)C(=O)NCC(CC)NC(C1CC1C(C)C)=O)OC C1(N(C(C2CC(CC)C2)=O)C)CN(C(=O)C=C2CCN(C)C2)CC1F Cn1nc(C(F)(F)F)cc1NC(C12CC1CN(c1ncc(Br)cn1)C2)=O c1(CNC(C)=O)cccc(C(=O)NCC(F)CNC(C2(C)CC=CCC2)=O)c1 c1(SC)nnc(CCCN(c2ccccc2)CC#N)n1C1CC1 CC1CS(=O)CCN1C(C1(CNC(C2CCC(CO)CC2)=O)CCCO1)=O C1(CNC(CCCN(C)C)=O)C(C)CCCN1C(C1CCCCC1)=O N1(C(c2c(C)oc(CO)c2)=O)CCCN(CCNC(C2(n3cncn3)CC2)=O)CC1 N1(C(c2nccc(CC)c2)=O)CC2CCC(C1)N2C(C1(C2CC2)CCOCC1)=O C1(CNC(CSCCC)=O)CC2(CCC2)CN1C(c1sccc1C)=O C(C)(C(C)(C)C(=O)NC1(c2cccs2)CC1)NC(C(CO)OC)=O CN1CC(C(=O)NC2CN(C(=O)C=Cc3ccc(=N)[nH]c3)CC23CC3)CCC1=O N1(C(c2c(C)cc(F)s2)=O)CCC2CC(NC(c3csnn3)=O)CCC2C1 c1(C(=O)Nc2nc(=O)s[nH]2)cc(=O)[nH]c2ccc(F)cc12 C1(C(=O)NC(C)CCCCNC(=O)CCC2CCCCC2)CCC2(C1)CC2(F)F N1(C(C2CCN(C(C)=O)CC2)=O)CC2CC(NC(c3c[nH]cc3Br)=O)CC2C1 c1(C(=O)NCCCCC(C)NC(CN(C(C)=O)C)=O)ccc(F)c(Cl)c1N CCCC(C)(CCC)C(=O)NCCNC(C1CN(C(C2C=CC=CC=C2)=O)C1)=O N1(CC(CC)NCc2ccccc2)CCCC(C)(C(N2CCC3CC3C2)=O)C1 c1(NC)c(C(=O)NCCN(C)C(c2c[nH]cc2C2CC2)=O)cccc1F C1(C(N2C(CCNC(Cc3ccn(CC)n3)=O)CCC2)=O)OCCN(C)C1=O c1(C(=O)NCC2(C(=O)Nc3c(C)cc(Br)cc3Cl)CC2)ccc2nc(O)oc2c1 c1(NC(C2C(NC(c3c(O)ccc(C)c3)=O)C2)=O)cc(Cl)c(Cl)cc1[N+](=O)[O-] C12(NC(=O)C3=COCCO3)CCCC1N(C(c1nc3ccccn3n1)=O)CC2 Cc1cc(C(=O)NCC2CCCC2NC(C2CCN(C)CC2)=O)n(C)n1 CC(N=c1nc2scnc2c(N(C)CCOc2ccncc2)[nH]1)C1CCOCC1 c1(C(=O)NCC2OCCN(C(CC3(C)CCC3)=O)C2)cccc2c1CCC2 C(=O)(CCC(C)OCC)N(CC(=C)Cl)Cc1nnnn1CSc1ccccc1 N1(C(C=C(COC)C)=O)CCCC(C)(C)C1CNC(=O)C(=O)NOC C1(O)(CN(C)C(C2(F)CCOC2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 c1(C(=O)NCC2C(NC(c3cnc(C(=O)OC)s3)=O)COC2)nn(C)c(N)c1C c1(CC)ccc(C(=O)NCC2(NC(c3cc(OC)n[nH]3)=O)CCOC2)cc1Cl C(=O)(CCC(=O)N1CC(NC(c2c[nH]cc2CC)=O)CC1C)N(CC)CC C1(C(C)NC(C2(C(N)=O)CC2)=O)CCN(C(c2ccc(CCF)cc2)=O)CC1 CC1(C)CC1(c1ccccc1)C(=O)NCCC1CN(C(c2ccoc2)=O)C1.C(=O)C1CC1 c1(C(=O)OC)ccc(OC(C)CCF)c(C)c1 N1(C(c2cnc(CC)s2)=O)CCCN(C(=O)CCCC(=O)N(C)C)CC1C Cc1cc(F)c(C(N2CCC(C)C(NC(=O)Cc3csc(S)n3)C2)=O)cc1F c1(C(=O)NCC2(F)CC(NC(C(=O)NC3CC3)=O)C2)ccc2nnc(O)n2c1 C1(O)(C(c2cccc(N3CCOCC3)c2)N2CC(C)(CC#N)C2)CCCCC1 C(=O)(CCC(C)C#N)N(CCC(=O)OCC)C1CC1 N12CCC(=O)N(C1=O)C(C1CCCCC1)CNC(=O)CCC2.C(=O)(NC)OC C1(C)(NC(C2C(OC)C2)=O)CCN(C(c2cc(C3CC3)on2)=O)CC1 N1(C(=O)CCn2cc(-c3ncoc3C3CC3)nn2)CC(C(F)(F)F)C(C(F)F)C1 N12CC3CC1CN3C(=O)C(Cc1cnc[nH]1)C2=O.c1(N(C)CC)cncn(C)c1=O c1(CC)ccc(C(F)(F)F)c(C(=O)OCC23CC(OC)(C2)C3)c1 C1(S(N)(=O)=O)(C(N(C)CC2CN(C(C3CCCCN3C)=O)C2)=O)CCC1 C1(CNC(Cn2ncc(CC)c2)=O)CCC2CN(C(=O)C(F)=CC3CC3)CC12 N1(C(CC(C)SC)=O)CCC(CCC(=O)NC2CN(C)CC2C)CC1 C1(CCNC(c2ccc(CCC)s2)=O)CN(C(c2cc(C)co2)=O)CCO1 N1(C(Cc2c(SC)cccc2)=O)CCC2(CC1)CN(C(=O)CC1CCOC1C)C2 C#Cc1cccc(C(=O)NC2CC(CCNC(c3ncccc3F)=O)C2)c1F c1(CCC)onc(C)c1C(N1CC(NC(C)=O)C(C)C1)=O C1(CNC(CCCC#C)=O)C(C)CCCN1C(=O)C(C)SCCCC N1(c2ccnc(NC(C)=O)n2)CCCN(C(=O)NC2CC(C)OC2=O)CC1 C1(NC(c2cc(CO)[nH]n2)=O)CCC2CCN(C(C3(C(F)(F)F)CCC3)=O)C1C2 N1(C(Cc2c(C)cccn2)=O)CC2CC(C1)CN(C(=O)CCCC(F)(F)F)C2 Cc1[nH]nc(C(N2CCCC(C3CCCN3C(=O)C=C3CCC3)C2)=O)c1Cl C1(NC(C(c2ccccc2)C)=O)CCC(NC(C2(C)CC(C(F)(F)F)C2)=O)C1 C1(CNC(c2ccncc2)=O)CSc2ccccc2O1 c1(-c2ccc(CNC(C(C)(O)Cn3cc(Br)c(=N)[nH]3)=O)o2)ccc(F)c(F)c1 C(=O)(NN=c1[nH]nc(-c2cccc(C(C(F)(F)F)OC)c2)s1)OC N1(C(C2(CNC(=O)C=CCCC)CC(=C)C2)=O)CC2CC(CO)C(C2)C1 c1(C(N2C(C#C)CCC2)C(=O)NCCCC)sc2ccccc2c1Cl N1(c2ncc(C)cn2)CC(NC(=O)C(CO)c2ccccc2)CC(C)C1 CC(C(=O)NCC(O)CC(=O)N1CC(S(C)=O)C1)C(C)(C)C c1(C(=O)NC(C)CNC(c2csc([N+](=O)[O-])c2)=O)c(F)cccc1[N+](=O)[O-] c1(C(=O)NC(C2CN(C(CC3(C=C)CCC3)=O)C2)C)cn2c(n1)CCCC2 C1(NC(c2cnc(CC)nc2)=O)CC2(C1)CC(NC(c1cc3n(n1)CCO3)=O)C2 C1(Nc2cc(N3CC(C)(C)C(CO)C3)ncn2)CC(c2ccccc2)=NO1 C(C(C)(COC)C(=O)NCc1cccc(NC(C2CCC(C)(C)OC2)=O)c1)OC N1(C(c2ccc(OC)cc2)=O)CCCC(NC(=O)CCc2cc(C)sc2C)C1C c1(C(C)NC(=O)NCC2CCC(CCO)CC2)nc2ccccc2[nH]1 N1(C(COC)=O)CCN(C(c2coc(NC(=O)C(F)(F)c3cncs3)c2)=O)CC1 N1(C(C(C)OCC#C)=O)CC2CCC1CN2C(c1c(C)[nH]c(C(N)=O)c1C)=O Cc1cc(C(N2CCCC(C)(NC(=O)C(O)C(F)(F)F)C2)=O)c2occc2c1 N1(C(C(C)C2CC2)=O)CC2(CCN(C(c3ccc(F)c(Cl)c3)=O)CC2)C1 C1(SC)CCC(C)(C)CC1c1nnc(-c2csc(C(C)C)n2)o1 n1(CC(=O)NC2CN(C(C3(SC)CC3)=O)CC2C)c(C)cc2ccccc12 C1(C(N)=O)CCCC(C(N2CC(O)(CCNC(=O)CO)C2)=O)C1.C1(C)CCOC1 C(=O)(CS(=O)(=O)C1CC1)NCC1OCCC(NC(CN(CCC)C)=O)C1 C(=O)(C(F)CC(C)(C)C)NC(C(=O)NC(C)CCCCCO)C1CC1 N1(C(CC(CC)N(C(c2c(CC)c[nH]n2)=O)CC)=O)CCN(C2CC2)CC1 Cc1cnc(C)c(C(=O)NCCC2CCCN2C(=O)CC2CC(C)=NO2)c1 c1(NC(c2n(C)cc(C(=O)OCC)c(=O)n2)=O)ccc(C(C)=O)c(C#N)c1 c1(C(=O)NCCN(C(c2cnc(CCC)s2)=O)CC)cc(OC)n(C)n1 CCC(C)(C(=O)O)N(C)C(c1cn(CC(c2cccc(Cl)c2)O)nn1)=O c1(NC(C2(CNCc3ccc(OCC)c(C)c3)CC2)=O)cc(F)c(C)cc1Cl C(C)(CCC(=O)NC1(CNC(=O)C(=O)NC(C(N)=O)C2CC2)CCC1)OC c1(OC)ccccc1CCC(N1CCOCC1CCNC(C1CCCCS1)=O)=O C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NCC(CC)(C)NC(=O)C(N)=O N1(C(C(C)NC(CCc2cc(C)[nH]n2)=O)=O)CCC(C2=NOCC2)C1 C(C(C(=O)NCC(Cl)Cl)C(C)C)NC(Cc1c(C)con1)=O N1(C(CCP(C)(C)=O)=O)CCN2C(=O)C(NC(c3cnc(=N)[nH]c3)=O)CC2C1 C(=O)(C1=NNC(=O)C1)N(CCNC(C1(c2ccon2)CC1)=O)CC CC1(C)CC(C(N2CC=CCC2)=O)CCN1C(=O)CCn1cccc1 N1(C(C)C)CCC2CCC(NC(=O)CCc3cn(C)nn3)C1C2 c1(N(CC(=C)C)CC(C)C)ncccc1S(=O)(=O)NCC12CCC(CC1)C2 c1(C(=O)OC)nn(C)cc1CNC(=O)NCC1(COC)CCOC1.c1(C)ccccc1 c1(C(=O)NC2CCC(NC(C3(CC=C)CC3)=O)CC2)cc(Cl)cc(F)c1N C(=O)(CN=c1[nH]c(=NCCC2CC(C)OC(C)C2)c2ccc(OC)cc2[nH]1)NCC C=C(C)C1OCCCC1C(=O)NC1CCC1NC(c1cc(Cl)cs1)=O CC1OCCC1C(=O)NCC(=O)NC1CC(C(=O)N(C)C)C1 Cc1c(F)ccc(NC(=O)CC2CCN(Cc3ccc(Cl)cc3F)CC2)c1Cl c1(CCC(=O)N(CC(CN(C(C)C)C)O)CC(O)CF)nc(C(C)(C)C)no1 n1(C(C)C)ncc2cc(NC(=O)CN=c3cccn[nH]3)ccc12 CS(=O)(=O)c1ccnc(NCC2CN(C(C3C=CCC3)=O)C2)n1 C1(CNC(C2N(C(CCc3n(C)ccc3)=O)CC=C2)=O)CC12CCOCC2 C(C1=CCN(C(c2nc[nH]n2)=O)CC1)NC(c1cncc(CC)c1)=O C1(NC(c2ncn(C)c2)=O)CCC(CNC(=O)CCC2NC(=O)NC2=O)CC1 C1(C)(C(N2CC3C(NC(Cn4ccc(C)n4)=O)(C3)C2)=O)CCCN(C)C1 C1(C)CC(C)(C)C(=O)O1.n12cc(cn1)CN1CC(C1)CNC2=O.CCS N1(C(C(C)=C(C)C)=O)CCC(C(=O)NCc2ccnc(O)c2)CC1(C)C N1(C(CCOCC(C)C)=O)CCC(F)C(NC(c2cc3n(n2)CCC3)=O)C1 C1(CN(C2CCOC2)C)CC2CC1CN(C(=O)CCOc1cccnc1)C2 C1(CC(=O)NCC2(O)CCN(C(COc3cc(C)on3)=O)C2)CCC(C)(C)CC1 c1(C(C)=O)cnn2c1CCCC2.C12(CNC(C3(C(N)=O)CCC3)=O)CN(C1)C2=O c1(NC(N(C(c2cnn(C)c2)CC2CCOC2)CC)=O)ccc(C)nc1N c1(C(C)(C)CCCN2CCOCC2)cccc(Br)c1.C12CCCN1C(=O)NC2=O CCC(C(=O)N1CCC(n2cccn2)(CNC(=O)C2=COCC2)CC1)C(C)C c1(OC)c(C(=O)NC2CC(C(=O)NC3CC(NC(N)=O)C3)C2(C)C)cnn1C C1(C(=O)NCCC2(O)CCN(C(=O)C(O)CCSC)C2)(CC)CC(C)(C)C1 N1(C(C2(CCC)CC(=O)C2)=O)CCC(F)(C(N2C(CO)CC2C)=O)C1 Cc1cccc(C2CC2C(=O)NCCC2CCCCN2C(c2coc(C)c2)=O)c1 c1(CCNC(=O)C(=O)NC23CCCC2NCC3)cccc(Cl)c1F N1(C(C2=CC(C)(C)C2)=O)CCn2ncc(CNC(c3cccc(Cl)c3F)=O)c2C1 C1(C(=O)N(O)Cc2cn(-c3ccc(Cl)cc3F)nn2)(OC)CCC(C)CC1 N1(Cc2cnc(C#N)cn2)CC2CCCC2(NC(C2CCC(C(C)C)CC2)=O)C1 C1(NC(Cn2nnc(C)n2)=O)C2CC3CN(C(c4[nH]c(O)nc4C)=O)C1C3C2 CC(Cc1ccco1)C(=O)N(C)CC1CN(C(c2ncoc2-c2ccon2)=O)C1 C(=O)(CCCC(=O)NCCCNC(C1CCCCN1C)=O)N(C)C C1(Cl)(C(=O)NC2CC(CNC(CC3CC(=C)C3)=O)C2)CC2CCC1O2 CCC(CC(F)F)C(=O)NCC1CCCN1C(=O)Cc1cccc(C(=O)OC)c1 N1(C(CCc2n(C)cnc2)=O)C2CCCC1CN(C(C1CCCCS1(=O)=O)=O)C2 Cc1nc(C2CCCOC2)sc1C(N1CC(CCC(C)Cc2cn[nH]c2)C1)=O N1(C2CCCC(OC)C2)CC(C(F)(F)F)OCC1C C1(C(N(C2CN(C(CCCOC)=O)C2)C)=O)Cc2ccc(F)cc2O1 Cc1[nH]nc(C(F)F)c1C(N1CCN(C(=O)CN2CCC(C)CC2)CC1)=O c1(NC(c2cncc(-c3c(C)cccc3)c2)NNC)nc(=NC2CCC(C)C2)[nH]c2c1SCC2 c1(C(=O)NC(CC)CN(C(=O)Cc2cnc(C)s2)C)c(N)cc(Cl)cc1F CCCCCCC(=O)NCC1C2CN(C(=O)C(C3CC3)N(C)C)CC12 C(=O)(C(C)CC(F)(F)F)NC1CCCN(C(c2nc(CCC)sc2)=O)C1 Cc1cnc2n1CCN(C(=O)C(c1ccnn1C)NC(=O)CCn1cnnn1)C2 N1(C(C2(C)COC2)=O)CCC2(CCCC2C(N2CCCC(c3ncc[nH]3)C2)=O)C1 Cc1ccc2nc(C(=O)NC3CN(C(=O)CN4CCC4C)CC3C)ccc2c1 c1(SC)cc(C)ccc1C(=O)NCC1CCCN1C(C1COC(=O)C1)=O c1(NC)cncc(C(=O)NC2(C(=O)N(C)Cc3c(C)noc3C)CC(F)C2)c1 C1(C(N2CCC(C)(CNC(c3cncnc3C)=O)C2)=O)(CC)CNC(=O)C1 CN1CCCC(C(=O)NCC2(CCNC(=O)CCCc3ccccc3)CC2)C1=O N1(C(C2CCN(CCCC)CC2)=O)CC2CC1CS2=O c1(C(=O)NC(C(C)NC(=O)NCCOCCOC)CO)ccc(OC)c(N)c1 C1(c2n(-c3c(CC)cccc3)nc(C3CC34CC4)n2)CC2(CCC2(OC)OC)C1 C1(CN(C(=O)CC2(C(C)(C)C)CCCC2)C)CCN(C(c2cn(C)cn2)=O)CC1 c1(CC)ccc(C)c(C(=O)NC(C2CCCC2)CNC(c2cc(Cl)no2)=O)c1 C1(C2CC2)(CNC(C(C)OC)=O)CCN(C(=O)C(C(C)(F)F)c2ccccc2)C1 c1(C(C)C)conc1C(=O)NC1COCC1n1cc(-c2csc(C3CC3)n2)nn1 n1(CC)ccc(CC(N2CCC(CN(C)C(c3csc(=N)[nH]3)=O)C2)=O)n1 C#CCC(C)(C(=O)N=c1ccn(C(C)CC)[nH]1)NC(C1C2CCC(C2)C1C)=O C1(C)(C(N2CC(C)(C(N)=O)C2)=O)CCN(C(=O)CC2(C(F)(F)F)CC2)C1 c1(C(=O)OCC)ccccc1COC(=O)C(F)(F)c1nc(C)cs1 C1(CN(C(=O)CCN(c2ccncc2)C)CC)CCCCN1C(=O)CCCF CCCCCCCCCC(=O)NCCC1CCC(NC(=O)Cc2cncn2C)C1 C1(C(C)CNC(=O)Cn2ccnc2)CCN(C(=O)C(C2(O)CCCCC2)F)CC1 C1(COC)(CNC(=O)CSCC#N)CCCN1C(=O)Cc1ccc(CO)cc1 c1(C(N(C(C)CNC(=O)C(C(C)O)N(C)C)CC)=O)ccc(=O)n(C)n1 c1(NC(=O)CC2CCCO2)ccc(C(=O)NC2CN(C(=O)NC)CC2C)c(Cl)c1 C1(O)(CNC(c2c(CC)nns2)=O)CCCN(C(=O)C(C)=C(C)C)CC1 C1(CC)(CC)CCN(C(=O)C(C)(C(C)C)NC(=O)C(C)N=[N+]=[N-])CC1 N1(C(C(=O)NCc2ccn(CCC(C)C)n2)=O)CCOC(C)(C(F)F)C1 C1(C(=O)NCCC(C)CCNC(=O)Cc2ccoc2)CC2CCC(C1)C2F c1(C(=O)NC(C2CCCCN2C(=O)C2=CSCS2)C)cccc[n+]1[O-] C#CCCCCC(=O)N1CC(NC(=O)C=CC(C)C)CC(O)C1 C1(C(N(CCOC)CCNC(=O)CSC)=O)CCSC(C)C1.C1(C(C)(C)C)CCCC1 C1(OC)(Cc2ccc(Cl)cc2)CCN(C(C2CCCN(C(C)(C)C)C2=O)=O)CC1 C1(O)(CCNC(C=CSC)=O)CCN(C(C2CC(C)CO2)=O)CC1 C(=O)(C(C)CC(F)(F)F)NCC(C)(C1CC1)NC(C(=Cc1ccncc1)C)=O c1(C(=O)NCC(F)CNC(C2CCCC2)=O)cn(CCO)c(=O)nc1O CC(CNC(=O)C(N1CCOCC(CN)C1)=O)CC(F)(F)F c1(SCCOC)cc(C(N2CC3CC2CN3C(=O)CC(C)(C)OC)=O)ccc1F N1(C(C2C(OC)C2)=O)CCC2OCCN(C(C3CCC3)=O)C2C1 CC1=C(C(=O)NC2C=CCN(C(c3oc(C)nc3C)=O)C2)CCC1 C1(NC(CC2(C=C)CC2)=O)CC2CCC1CN2C(c1cnc(OC)nc1C)=O C1(C(N2C(SCC=O)CC2)=O)C(O)CC1O CC1(C)CCC(C)(C)N(C(C2CCC(CC(F)(F)F)CC2)=O)C1 c1(OC)cccc(NC(=O)NC2CC=CCC2C(=O)N(C)C)c1F C(CCC(=O)N(CCCOCCO)CCO)C1C(C)C1.C1CC(=O)N1 CCC(O)C(C)(C)C(=O)N1CCN(C(c2ccnc(S)c2)=O)C(CF)C1 N1(C(CS(=O)(=O)NCC)=O)CCN(C(=O)CCC2CCOC2)CCC1C CC(C)C(C(C)NC(c1ccc(C(F)F)s1)=O)NC(c1ccnc(C2CC2)n1)=O N1(C(C(C(COC)C)C)=O)CCCN(C(=O)Cc2cc(OC)ccc2Cl)CCC1 C1(OC)(CNC(C2CC2C(C)(F)F)=O)CCN(C(C2CC2C(F)(F)F)=O)C1 C1(NC2CCN(C3CCCN(C(=O)OC(C)(C)C)C3)C2=O)CCN2CCOCC12 CC1(C)NC(=O)CC1C(N1CCCC(C)(CNC(C2CC2c2ccco2)=O)C1)=O N1(C(C2CC(C#C)(O)C2)=O)CC2CCC(CNC(c3ccnc(C)n3)=O)C2C1 CCC(CC(=O)NCCCCC1CN(C(=O)CNc2nccs2)C1)C(C)C N1(C(C(=O)NC2(C)CC2)CCc2ccco2)CCCC(CO)(CO)C1 c1(C(N2CCC(C(N3CCOC(CF)C3)=O)(OC)C2)=O)ncc(F)cc1F C(C(C)(COC)C(=O)N1CCC(C(C)C(=O)NCC2(CCO)CCC2)C1)OC CCC(CC(=O)N(CC(C)(C)CNC(C1CC(=C2CCC2)C1)=O)CC)SC C1(NC(COCC=C)=O)COC2C(NC(=O)Cc3c(F)cccc3Cl)COC12 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CCC2(C(NCc3cccc(C#N)n3)C2)CC1 C(CCC1CC1)(C(=O)NCc1ccc(O)cc1)NC(c1cn(CC)nc1)=O Cc1nn(C)c(Cl)c1CNC(C1CC1NC(=O)CCOc1cccc(F)c1)=O N(C(=NCCOC1CCSCC1)NCc1ccccc1)CC1(C)CCC1 CCC(C(C)C)C(C(=O)NCC(F)F)N1CCC(c2nc3cccc(Br)c3o2)C1 c1(C(N2CC(C)(CCC(=O)N(C3C(C)C3)C)C2)=O)cc(O)cc(F)c1 c1(N2CC(C)(NC(=O)C(=O)Nc3ncc[nH]3)C2)nccc(S(C)(=O)=O)n1 N1(C(c2ccn(CC)n2)=O)CCC(CC)(NC(=O)C(c2cnn(C)c2)C)CC1 C(=O)(CCCC(C)=O)NC(C1CCCN1C(=O)COCC1CCCO1)C C(=O)(CCCC(F)(F)F)NC(CNC(c1c(C)onc1Br)=O)(C)CO C1(C(N2CC(OCC(=O)N(CC(C)O)CC(C)O)C2)=O)CC(C)(C)CCO1 C1(CNC(=O)Cc2cncnc2)CC2CCC(C1)N2C(=O)C1=C(Cl)CCCC1 C1(C2CCC2)(C(=O)NC2C(OC)CN(C(=O)C(C)(C)COC)C2)CC1(F)F Cc1ccc(CCC(=O)NCCC(O)CNC(=O)C=CC2CCCO2)cc1 C(=O)(C#CC1CCOCC1)N(C1(C(N(C(C2CCCC2)C)C)=O)CCC1)C1CC1 N#CC1CCCC(C(N2CCCC(C(=O)NC3CCC3)C2)=O)C1 c1(C(C(N2CCCC(CNC(CC(C)OC)=O)C2)=O)(F)F)ccc(=O)n(C)c1 Cc1cc(CC(=O)N(C)CC2(O)CCCN(C(=O)C(F)=CCCF)C2)ccc1Cl N1(C(C(C)OCC=C)=O)CCC(O)(CNC(c2cccc[n+]2[O-])=O)C1 N1(C(Cc2ccc(C)nc2)=O)CCN(C(c2n[nH]c(C)c2Cl)=O)CC1C c1(C(N2CCCC(N(C(C(C)NC(=O)NC)=O)C)C2)=O)cc2n(n1)CCNC2=O c1(CCCC(=O)N2CC(=C(CNC(C3CC(C)(F)C3)=O)F)C2)ccc(F)c(F)c1 Cc1ccc(CCC(=O)NCCOCCNC(C2CCC(C(N)=O)O2)=O)cc1Cl CON1CCC(C(=O)NC2CN(C(=O)CSC(C)(C)C)CCC2C)CC1 C1(CNC(c2c(COC)noc2)=O)(CO)CCN(c2ncnc(C)c2F)CC1 CC1CCN(C(=O)C=Cc2cnc[nH]2)CC1NC(=O)C=CCN1CCCC1 c1(C(N(C2CCN(C(Cc3c(C)n(C)cn3)=O)CC2)C)=O)ncc([N+](=O)[O-])n1C c1(CN(C(C(C)(C)c2ccccc2)=O)Cc2cnn(CCO)c2)ccccc1F C(C(F)C(=O)NCC(CSC1(c2cccnc2)CCCC1)OCC(=NO)OC)OCC C1(C)(C(N(CCCCN(C)C(C2CC2(Cl)Cl)=O)C)=O)CCCNC1=O C1(NC(CCC(=O)NC)=O)CCC2CN(C(c3ccn(C)c3)=O)CC2C1 N1(C(C(C)OC)=O)CCC2C1CCN2C(=O)C(c1ccccn1)Oc1ccccn1 C12(C(=O)NC3CC(NC(c4c(OCC)scc4)=O)C3)CC(CO1)C2(C)C c1(C(N2CC(COC)N(C(=O)CCS(C)=O)CC2)=O)cc2c(C)ccc(F)c2o1 Cc1cc(CCC(=O)NC2CCN(C(=O)OC(C)(C)C)C2C)nn1C C=C(Br)CC(C)(C)C(=O)NCC1CC1NC(c1ccn(CC(C)C)n1)=O CC(C)(CNC(=O)C(c1ccoc1)NC(=O)CC1CCCC(=O)N1)C(N)=O C1(NC(C(CC=C)C)=O)CC2CN(c3cc(C)c([N+](=O)[O-])cn3)CC2C1 n1(CCC)cc(C(N2CCC(N(C(=O)C(C)CC(C)C)C)C2)=O)c2ccccc12 c1(C(=O)NCC2C(NC(C(C)c3cccs3)=O)COC2)cnn(C)c1Cl c1(C(N(CCN(C(c2c(CCC)nsc2N)=O)C)C)=O)cccc2cncn12 N1(C(C(CCCC)N(C)C)=O)CCC2(CCN(C(c3ccnnc3)=O)C2)C1 c1(C(N(CCN(C(CCC=C=C)=O)CC)CC)=O)cnc2c[nH]nc2c1 N1(C(CCC=C)=O)CCOC2(CCN(C(c3cnc4cc(C)nn4c3C)=O)C2)C1 c1(C(=O)NC(C(=O)OC)C)n[nH]cc1CNC(=O)CCOC1CCCC1 C(C)(C)(CC(F)C(=O)NCC(C)(O)COC)NC(C=C(CCC)CCC)=O C1(CCNC(=O)Cc2cccnc2)CC(F)(F)CN1C(=O)C(C1CC(F)(F)C1)O c1(OC)cc(C(C)C)cc(NC(=O)C(C)(C)O)c1C(C)C C1(C(=O)NCC(CC)NC(c2cc(O)nn2C)=O)(N(C)C)CCCOC1 CCCC(O)CC(=O)NC1CCN(C(=O)Cn2ccc(C)n2)C1 CC1CCC(=CC(N2CCOC(CN(C(=O)CC3CCCCO3)C)C2)=O)CC1 N1(C(c2cc(C)cc(C)c2)=O)CCCCC12CN(C(C1(C)CCCC1(F)F)=O)C2 c1(C(N2CCN(C(C(C=C)O)=O)C(CF)C2)=O)ccc(S(=O)(=O)NC2CC2)o1 n1(CC)ncc(C(=O)NCC2CC2CC(=O)NC2(CC)CCOCC2)c1Cl N1(CCC)C(=S)NC(c2cc(OC)c(F)cc2F)C2=C1C1(CCC1)NC2=O N1(C(C2CCN(C)C2)=O)CC2CCCC2(C(=O)NCc2nccs2)C1 C(C(=O)NC1(CNC(=O)C2=CSCCO2)CCC1)(C(C)(C)C)OC O=S(=O)(c1nc(N2CCC3(CCCCC3)C2)ccc1Br)N1CC2CC2C1 N1(C(c2c(C)c(Br)no2)=O)CCOCC(NC(C2(C)CCCS2)=O)C1 N1(C(COCC(C)C)=O)CCC(n2cccn2)(CNC(=O)Cc2cncs2)CC1 N1(C(CCC2CCCN(C(CCC(=O)NCCC)=O)C2)=O)CCCC(C)(O)CC1 c1(CC(=O)OCC)c(C)[nH]c(C(=O)C(F)(F)c2ccsc2)c1C N1(OC(c2cn(Cc3ccc(OC)cc3)nc2)=O)CCCC12CCNC2 CCC(CC(=O)OC)NC(c1oc(CNC(=O)Cc2ccn(CC)n2)cc1C)=O c1(C(N2CC(CNC(c3cc(C)no3)=O)N(C)CC2)=O)cc2nnn(C)c2s1 C#Cc1cn(C)nc1C(N1CCOC(C(=O)NC(c2ncccc2F)C)C1)=O C1(NC(C=C(C)Cl)=O)CCN(C(c2ccc(F)cc2)=O)C(C)C1 c1(C(=O)NCCC2(CNC(c3n(CC)nnc3)=O)CC2)cc2c(s1)CCCC2 CC1CN(C(C2CCCCN(C(=O)CCN(C)C)C2)=O)Cc2ccc(Cl)cc21 C(=O)(C1=CC(O)C(NC(=O)CC2CC3CC3C2)C1)NCCNC(=O)CO C1(N(C(CCC#CC)=O)C)CCN(C(c2ccc(C)cc2Cl)=O)CC1C c1(OC)cc(C2(NCc3cnn(C)c3-c3ccncc3)CC2)cc(F)c1F C(CCC(C)C)(C(=O)NCC1(C(F)(F)F)CC1)NC(C(CC)C)=O C1(C(=O)NCC(O)C(F)(F)F)CC2CCC(C1)N2C(C1(F)CCCCC1)=O c1(CN2CC(NC(CC(CC)O)=O)C(F)(F)CC2)ccc(C)cc1[N+](=O)[O-] C=CCCCCCCC(=O)NCCOCCC(=O)NCCc1cnc(C)[nH]1 C(=O)(C(C)(C)CNC(=O)C(C)CN(C)C(c1cncc(C)c1)=O)NCC C(=O)(C1CCc2ccccc21)N1CCC(O)(C(=O)Nc2cncnc2Cl)C1 CCCCCCNC(C1(NC(=O)CC2C=CCCC2)CC(F)C1)=O c1(C(N(C(C)CNC(=O)CCCc2nncn2C)CC)=O)cc(Cl)cnc1O N1(C(c2c(C)cc(CC)o2)=O)CCCC(CC)(NC(=O)Cc2ccncc2Cl)C1 c1(CNC(C(CC)SC)=O)cncc(NC(=O)C(c2ccccc2F)OC)c1 Cc1ccc2sc(C(N3CC4CC(NC(=O)CCCC(C)C)CC4C3)=O)cc2c1 C(=O)(C1=C(Cl)CC1)NC1CC(F)(CNC(=O)CC(C2CC2)C2CC2)C1 N1(C(C(CNC(=O)NCC#C)O)=O)CCC(C(=O)NCC=C)(SC)CC1 C#Cc1cccc(NC(C)C(N2CCN(C(=O)C(F)n3cccn3)CC2)=O)c1 C1(NC(COCc2cc(C)on2)=O)CCC12CN(C(c1cc(Cl)ccn1)=O)C2 N12CCCCC1C(=O)NC(=O)C(C)n1cc(nn1)C2.C(=O)(C(F)(F)F)OC(C)C O=C1CC(=O)NC(C(=O)NC2CC(C(F)C(=O)NCc3ccncc3Cl)C2)C1 Cc1cc[nH]c1C(=O)NC(c1ccccc1)C(=O)NC1COC(C(F)F)C1 c1(CNC(=O)C(N2C3COCC2C3)c2cn(C3CCOC3)nn2)ccccc1F C1(CNC(c2cocn2)=O)C(C2CC2)CCN1C(c1csnc1Cl)=O C12(CNC(c3ccc(C)cn3)=O)CCC1CCN2C(=O)CN1CCC(CO)CC1 C=CC1CN(C(=O)C(C)NS(=O)(=O)CCCC)CC1NC(c1ncccc1C)=O c1(CC)cccc(CC(=O)NCCN(C(c2cc(C)c(Br)o2)=O)C2CC2)c1 c1(C(N2CC(NC(Cc3c(C)noc3)=O)C(C)CC2)=O)cnc2cccc(C)n12 C(=O)(C1CCCc2nc[nH]c21)NCC1(F)CC(CNC(=O)CCOC2CC2)C1 CC1C(=O)CC1C(=O)NCC(O)CNC(C1CCCN1C)=O C1(CNC(Cc2ccn(C)n2)=O)CC2COCC2N1C(c1ccncc1)=O Cc1ccc(C(N2CCC3CN(C(=O)Cc4cncs4)C3C2)=O)c2c1CCC2 C(CCC(=O)N1CCCC1CC(=O)NCC(C1CC1)SC)OC C1(C(=O)NCCC)CC(O)CN1C(=O)C(c1ccccc1Br)NC(=O)OC N1(C(Cn2ccc(OC)n2)=O)CC2CN(C(c3cc(C)c(O)nn3)=O)CC2(C)C1 c1(OC)ccccc1C(=O)NC(CNC(=O)C=C(C)C1CC1)CC(C)C.C(F)F C(CCC(O)C(=O)NCCCC1(C)CC1)NC(C(CCC)OC)=O N1(C(C(CC)CC)=O)C2CCC(C2)C1CC(=O)NC1C=CC(CO)C1.C(C)C Cc1nnn(CC(=O)NCC(C2CCCC2)NC(C2(O)CCOC2)=O)n1 C1(C(=O)NCC2CC(NC(CCC(C)C)=O)C2)CN2CCN1CC2C C1(C(=O)NCC(C)NC(=O)C=CC2CC2)CNC(=O)C1 c1(OC)ccc(CC(=O)NC(C)CNC(=O)CC2CC(C)(C)CCO2)c(C)c1 c1(C(N2C(CO)CC(NC(C3CCCS3)=O)C2)=O)c(Cl)ccc2c[nH]nc12 C(=O)(C(O)CCCc1ccccc1)NC(CC)CNC(C1(N(C)C)CCC1)=O FC(F)(F)CC(c1nnnn1Cc1cccs1)NCCCSc1cnc(Cl)s1 C1(C2N(C(C3C(C)C3)=O)CCC2)CCN(C(=O)CCOC(C)C)CC1 CC1(C)CCCOC1NC(N1CC(O)(c2cn(-c3cc(Cl)ccc3F)nn2)C1)=O C1(C(=O)Nc2ccncc2F)CCN(C(N(C(CC)C)C)=O)CC1 C(=O)(C1=CCCCO1)NC1CN(C(=O)C2=CCCC2)CC1CO C(=O)(C1=C(C#N)CCC1)NCCc1c(C(N2CC(CC)OCC2C)=O)c[nH]n1 c1(OCC)cccc(CC(=O)NC2CCCC(NC(c3n[nH]c(CC)n3)=O)C2)c1 C1(CC)COCCN1C(=O)C(C)NC(=O)C1=CCSC1 N1(C(C(C)C)=O)CCC(N(C(=O)COc2ccc(Br)cc2Cl)C)C(C)C1 Cc1ccc2[nH]c(C(=O)NC3(C)CCCN(C(c4sc(F)cc4C)=O)C3)cc2c1 CC(=O)CCCC(C)C(=O)NC1(C(N2CCC3(CCC(O)C3)C2)=O)CCCCC1 c1(CC)cnc(O)c(C(=O)N(C)CC2CCN(C(C3CC3C)=O)C2)c1 C1(C#N)(C(=O)NCC(N(C(C2C(=C)CC2)=O)C)C2CC2)CC12CCC2 C1(C(N2C(C(=O)NC)CCC2)=O)CC(C2CNC2)C1 n1(CC(=O)N(CC(CNC(CC(C)(C)OC)=O)C)C)cccc(C)c1=O C1(C(=O)NC(C)C(C)NC(=O)C=C2CCCC2)CCC(OC(F)(F)F)CC1 N1(C(C(Br)=C(C)C)=O)CCC(CNC(=O)C(C)Cn2cccn2)CC1 c1(C(N2CCC(C(C)N=c3nc(C(C)(C)C)[nH]s3)C2)=O)ccc2ccncc2n1 C1(NC(C2CCC(CC)CC2)=O)CCC12CCN(C(=O)Cc1ccsc1C)CC2 N(C1CCCc2c1cnn2OCC#C)C(=O)OC(C)(C)C CC1=C(C(=O)N2CCSCC2C(N2CCNCC2)=O)S(=O)(=O)CCO1 CCC(CC)(CO)C(=O)N1C2CCC1CN(C(=O)CC13CCCC1C3)C2 C(C(C)(F)C(C)(C)F)n1cc(CNC(C2(C)CC3(CC3)C2)=O)nn1 c1(C(C(=O)NCCCC(C)C)N(CC(=O)OC)C(C)C)ccc(C(F)F)cn1 c1(COC)ccc(C(=O)N(C2CCN(C(C3C=C(C)CS3)=O)C2)CCO)s1 CC(C)CCCC(C)C(=O)NCC(C)(C)C(=O)NC(C1CCOCC1)C C1(C(N(C)CC2(NC(=O)C=Cc3cncnc3O)CC2)=O)C2CCC1(C)C2(C)C C(=O)(CCC(C)CN(C)C)NCC1(CN(C(C(C)SC)=O)C)CC1 CCC(CCC(=O)N(C)CCOCCC(=O)N(CC(O)CC)C)OC n1(CC)nc(C)c(C(=O)NCCC2CCCCN2C(=O)C=CC2(C)COC2)c1C C1(NC(c2c(CC(C)C)nc(C)s2)=O)CC(O)CN(C(=O)COC(C)C)C1 C(=O)(C1COc2ccccc21)NCC1CN(C(CS(=O)(=O)N(C)C)=O)CC12CC2 Cc1ccc(F)cc1-c1cn(CCCC(=O)N(CC(C)C)CCO)nn1 C(C1CC1)(C1CC1)=CC(=O)NCC1(NC(C(C)CN2CCOCC2)=O)CCC1 Cc1cccc2c(C(=O)NC(CNC(=O)C(N)=O)CO)coc12 CC1CN(C(=O)CN(CCCF)C)CCN1C(C)=O.C(C)(C)(C)OC=O N(C1CCCc2ccoc21)C(C1=CCN(C(CCC=CC)=O)C1)=O c1(C(=O)NC2CCC2NC(c2cccc(C3CC3)c2)=O)ccc2oc(S)nc2c1 CC(CC(C)(C)C)C(=O)N1CC(C)(C)CC1CC(N1CCOCCC1C)=O C(=O)(C(C)(C)CS(=O)(=O)N1CC(N=[N+]=[N-])CC1C(=O)OC)OC C1(NC(CC(C)OC)=O)CCN(C(c2cc(C3CCC3)[nH]n2)=O)CCC1(F)F n1(CC)nc(C(N2C(C(=O)NC3CCOC(CC)C3)CCC2C)=O)cc1C C12(NC(CCCc3onc(C)n3)=O)CCCC1CN(C(c1cc(C)c(C)o1)=O)C2 CC1CC(NC(c2cc(C(C)(C)C)nn2C)=O)CN(C(c2cccnn2)=O)C1 C(CNC(N)=O)(CCNC(C1(SC)CC1)=O)OC C1(Cn2cc(C(C(=O)NCC(C3CCOC3)NC)(C)C)nn2)CCCC(=O)C1 N1(C(CCC=CCC=C)=O)CCC2(CC1)CN(C(=O)Cn1cccc(C)c1=O)C2 Cc1cc(NC(=O)C(O)CCNC(C2(C)CCC(=O)NC2)=O)cnc1O C(=O)(C(O)CC(C)(C)C)NC12C(CN(C(c3c(C)nc(CO)s3)=O)C1)C2 C1(C#N)(C(=O)NCC2C(CC(=O)N(C)Cc3n(CC)ccn3)C2)CC1(C)C CCCCC(CC)C(=O)N1CC2(C(=O)NC(C)(C)CC3CC3)CC1CCO2 N1(CC(=O)NC)CC2CC(NC(C3CC4(CCC4)CN3C)=O)CC1C2.C1CC1 CCCCC(CNC(=O)CC(C)n1cc(Br)cn1)NC(=O)CCc1nc[nH]n1 Cc1[nH]c(C#N)cc1C(N1CCC(CF)(NC(c2nocc2Br)=O)C1)=O C1(O)(CC(N2CCC(CN3CCC3)CC2)=O)CCN(C(=O)CC(O)C2CC2)CC1 c1(OC(CC)CC)ccccc1C(N1CC(NC(c2cc[nH]c2C)=O)C(C)C1)=O N1(C(c2ccc(NC(c3ncc(C)c(Br)c3)=O)nc2)=O)CC2(CNC(=O)N2)C1 C1(CNC(C2C(C)C2(F)F)=O)CCCC(NC(=O)CN2CC3CC3C2)C1 Cc1ccn(C)c1C(N1CCCC(CN(C)C(c2cc(Cl)ccn2)=O)C1)=O O=C(C1=CC2CCC(C1)C2)NCC1CCC(NC(c2cn[nH]c2)=O)C1 Cc1cnc(C(N2CCOCC2c2cn(Cc3cccs3)nn2)=O)c(Cl)c1 C1(C(N2C(CO)CC(NC(COCC=C)=O)C2)=O)CN2CCC1(C)C2 c1(C(N)=O)ccccc1C(N1CCC(C(=O)NCC(CO)CO)C1)=O C12(C(=O)NCCOCCNC(c3c(C)nsc3C)=O)CCCN1CCC2 N1(C(c2c(NCC)scn2)=O)C2CCC1CC(NC(=O)CCCN(C)C(C)=O)C2 Cc1cc(C(=O)N(CCCC(=O)NC2CCN(C(C)(C)C)C2)C)c(C)n1C CC(N=c1[nH]c2c(c(=NCc3cncs3)[nH]1)SCC2)c1ncnn1C c1(C(=O)NC2(C)CCCN(C(C3(CC4CCC4)CC3)=O)C2)cnn2cnnc2c1 c1(C(N2CCC(CCNC(C(CC)OC)=O)C2)=O)ccc(OC2CC2(F)F)cc1 c1(C(=O)NC(C2CCN(C(c3ccc(COC)cc3)=O)C2)C)cnc(Cl)cc1N C1(NC(C(CC)=CC)=O)CC2CCC1CC2NC(=O)COCCCC(C)C N1(C(CCCN(C(C)=O)C)=O)CC(NC(=O)C(C)CN(C)C)CC(C)(C)C1 C(C1=NOC2CN(C(=O)C=Cc3nccs3)CC12)NC(c1nncs1)=O CCC(CC)C(=O)NCC1CCCN1CC.c12ccccc1CNC2=O C1(CC)(CNC(C2C(NC(=O)CC3CCOC3C)C2(C)C)=O)CCOC1 c1(NC(N)=O)cocc1NC(=O)CC1CCN(C(=O)CC2CC=CC2)C1 C1(O)(CN(C(=O)CSc2cccc[n+]2[O-])C)CCCN(C(=O)Cc2cscn2)C1 C(C(O)CC(C)(C)C)NC(C1(CC)CN(C(COCCC#C)=O)C1)=O C1(NC(c2cc(OC)n(C)n2)=O)CCCC(C(=O)NC(CO)(CO)CO)CC1 C(N=c1[nH]c(=NCCN2CCP(C)(=O)CC2)[nH]c2c1COC2)c1ccc(C)nn1 C1(C(=O)NCC2C(NC(c3ccc(-c4ccccc4)o3)=O)C2)CC2(C1)CC(O)C2 Cn1cc(C2CC2C(N2CCCC2c2nc(CCNC=O)no2)=O)cn1 N1(C(C(CCC)OC(N)=O)=O)C2CCC1CN(C(C1CC1(C)C(=O)NCCCC)=O)C2 c1(C(CC(=O)NC)NC(N2CCC(CC(C)(C)C)C2)=O)ccc(O)cc1 C1(NC(C2(OCC)CC2)=O)CCN(C(c2cccc(C#N)c2)=O)CC(C)(C)C1 c1(CN2CC(NC(c3ccc(I)c(Cl)c3)=O)C(F)C2)csc2ccccc12 C(=O)(C1CCCn2cnnc21)NC1CCC(C)(C)C1.C1CCN1C c1(SC(C)C)cc(C(N2CCCC2C(C)NC(C2(CCN(C)C)CC2)=O)=O)sn1 C1(C(=O)NCc2c(SC)c(F)ccc2)CC2COCC(C1)C2 O=[N+]([O-])c1c(Br)cc(-n2nnnc2O)cc1Br.C12(CO)C(CC1CCO)OCN2 c1(C(N2CCC(C(C)C(=O)NCc3cscn3)C2)=O)ccc(O)c(F)c1 C1(C(=O)O)(NC(C2(OC)CCOC2)=O)CC2CC(O)C(C1)N2C c1(NC(=O)NCc2ccc(OC(F)F)nc2)ccc(-c2cscn2)cc1 C1(CNC(C2(C)CC(C)C2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1C N1(C(CCS(=O)(=O)NC)=O)CCC(C)(C)C(C(N2CCCC2CO)=O)C1 C(=O)(C(C)(C)C(C)(C)O)NCC(CN(C(C(C)CC(N)=O)=O)C)(C)C C(CCC(=O)NC(C1(O)CN(C(=O)C=CCF)C1)C)SC C1(NC(c2c(C)con2)=O)CC2CC(C1)N(C(c1ccnc3ccnn13)=O)C2 c1(C(=O)NCC(CC)NC(C2C3CCC(F)(F)C23)=O)cc([N+](=O)[O-])cnc1N C(CC(O)CNC(=O)CSC(F)F)NC(C(c1cccs1)SC)=O C1(OCCNC(c2cnc(Cl)[nH]2)=O)CCN(C(=O)CC2CCC(=O)NC2)CC1 CC(=Cn1ccnn1)C(=O)NCCC1CN(C(=O)CC2CCCCN2C)CC1C C#Cc1cccc(NC(=O)C(N2CCOCC2CNC(=O)CSCCOC)=O)c1.C(C)=CC C1(SC)CN(C(C2CCCCN2C)=O)CC1NC(c1ccc(C(N)=O)cn1)=O N1(C(C(SC)SC)=O)CC2CC(C1)CN(C(=O)C(C(C)C)n1cncn1)C2 C1(NC(c2cc3cnccc3o2)=O)CCN(C(C2(C(F)F)CC2)=O)C12CCCC2 CC1CC(=O)NC1C(=O)NC1(CCCNC(c2[nH]c(O)nc2C)=O)CC1 C1(OC)CCCN(C(C(=O)NC2CCC(F)(F)CC2)C(C2CC2)OC)CC1 C(=O)(C(O)C1=CCCCC1)NCC(CCCC)NC(c1cccc(Cl)c1F)=O N(C1CCC(NC(=O)C(CC)(CC)OC)c2ccccc21)C(CSCCC)=O C1(C(=O)NCC(C2C(CC(=O)OC(C)(C)C)CC2)(C)C)CCC(C#N)CC1 N1(C(C(C)OCCC(C)C)=O)CCC(C2(NC(C3CC4(CC4)CO3)=O)CC2)CC1 N1(C(C2(C)CCCCC2)=O)CC2CC(CC(=O)NOCC=CCl)C(C2)C1 C1(C(=O)NCC(CO)NC(C2OCCO2)=O)(OC)CCCOC1 Cc1ccc(C=CC(=O)NC2CCCC(CN(C(=O)Cc3ccccc3)C)C2)o1 C1(CC)CN(C(c2ccc(C#N)[nH]2)=O)CC1NC(c1nc(Cl)sc1C)=O c1(C(=O)NC2CCN(C(CC(C)C3CC3)=O)CC2O)cc(=O)n(C)cc1Br C1(CN(C(C(C)C#N)=O)C)CCCN(C(=O)COCC(F)F)C1 c1(NC(N2C(C)(CNC(c3c(OC)cccc3)=O)CCC2)=O)oc(C)nc1C#N C(CCCCC(=O)NC1CCCC1CNC(=O)CCc1cscn1)OCC C1(N(C(C2C(COC)CC2)=O)C)CN(C(c2c[nH]c(C#N)c2)=O)CC1O c1(NC(N(c2ccccc2F)CCC)=O)ccc(C(F)(F)C(=O)OC)cn1 c1(NCc2cc(C)[nH]n2)nc(N2CCC(N(C)C)C(C)C2)nc2c1cnn2C NC(=O)C1=NOC(CNC(=O)C(C2CCCO2)NC(c2csc(Cl)n2)=O)C1 N1(CC(N2C(C(C)NC(C(CC)CCOC)=O)CCC2)=O)CCCCCCC1=O C#CCCCCC(=O)NCC1C2CC1N(C(=O)CCN(c1ccccc1)C)C2 c1(C(C(=O)NN2CCCC2)(F)F)c(F)cccc1Cl.c1(C(C)=O)ccccc1 Cc1ccc(C)c(-n2nc(C)c(C(=O)NCCn3cc(C4(C)CC4)nn3)c2Cl)c1 c1(CC(=O)NCC(C2CC2)NC(C=CC2N(C)CCC2)=O)ccc([N+](=O)[O-])c(N)c1 CN1CC(C(N2CCOCC2C(=O)NCCC2CC(C)(C)C2)=O)CCC1=O C(N=c1cc(C)[nH]c(=NCCNC(=O)NC(C)(C)C)[nH]1)C1(OCC)CCC1 C1(O)(C(C)NC(Cn2c(C)nnn2)=O)CCN(C(c2cccn2C2CC2)=O)C1 C1(OC)CN(C(c2cn(CCO)nn2)=O)CC1C(N1CCCC1CF)=O C1(OCC(=O)NCCN(C)C=O)(CSC)CCCCC1.C1(CCC)(CC)CC(=O)C1 C1(NC(C2(C#C)CCC2)=O)CCOC2(CCN(C(C3CCCO3)=O)CC2)C1 c1(C(N2CC3CCC2CN3C(C2CCC(F)C2)=O)=O)nc2ccc(Br)cc2s1 c1(C(=O)NCC2C(C)CN(C(C3C=CCS3)=O)CC2)cnn2ccccc12 C(C(C(=O)N(C)Cc1cnc(C)s1)NC(=O)Cc1cnnn1C)OC c1(CC)cnccc1C(=O)NCC1C2CN(C(=O)CNS(C)(=O)=O)CC12 C1(CC(N2CCC(C(C(=O)NCC3(C(F)(F)F)CC3)F)C2)=O)CCCCCC1 C(=O)(CC(C)(C)C1CC1)NC1(C)CC(NC(CCNC(COC)=O)=O)C1 N1(c2n(C)c(C(c3nc[nH]n3)=O)nn2)CCC(C2CC2)C1Cc1ccco1 C(CCCCCC(=O)N1CC(SC(F)F)C1)NC(N1CCCCCC1)=O C1(OC)CCC2(CCN(C(=O)C(=O)NCC3CCCC4(CCC4)O3)CC2)O1 CCC(C)(CNC(c1ccsn1)=O)C(=O)N1CC(O)C(O)C1 C12(C(N3CCC(C(C#C)C)CC3)=O)CC(CO1)N(C(C1(CC)CC(C)(C)C1)=O)C2 CC1C(C(=O)NCc2nc(N(C)C)n[nH]2)CCCN1C(c1cccnn1)=O CC(C#N)C(=O)N1CC(N(C)C(c2cc(C3CCC3)no2)=O)C1 C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(=O)CC(F)(F)F)C2(CCC2)C1 C1(NC(CN(C)CCO)=O)CCCCC12CCN(C(=O)Cc1cnccc1Cl)C2 C(CNC(c1ccccc1-c1cc[nH]n1)=O)(CC)(CC)NC(C1CC(OCC)C1)=O c1(OC)c(C(=O)NCC2(NC(C3CCC(CC(C)C)O3)=O)CC2)ccnc1F C1(CCNC(c2ccc(OC)s2)=O)CC2CCC(C1)N2C(C1CC2(CC2)C1)=O C1(CC)CN(C(c2cnc(C(C)=O)s2)=O)CCN1C(=O)Cc1ccn(C(F)F)n1 c1(C(=O)NC(Cc2cn[nH]c2)C(=O)N2CCC(OCCOC)C2)cncc(CO)c1 CC1CCC(NC(C2(C#N)CC2)=O)CN1C(c1cc(C(F)(F)F)n(C)n1)=O N1(C(CCCCOCC)=O)CC(C)(C)OC2(C1)CN(C(C1CCC(F)CC1)=O)C2 C(=O)(C(C)(F)C(=O)NCCC(C)(C)NC(=O)COC1CCCC1)OC c1(C(CNC(c2n(CC#C)cnn2)=O)NC(=O)CC(C)OC)cccc(OC)c1 c1(N(CCOC)CCSC2CCCO2)nccc(=NCCC#N)[nH]1 c1(C(c2n(C)nnn2)NCC2C(C)(C)C2(C)C)csc2ccccc2c1=O C1(C(=O)NCCCCCCNc2c(C(N(C)C)=O)cncc2)CCCCNC1=O n1(CC(F)(F)F)ccc2cc(NCC3COC4(CCC4)C3O)ccc12 c1(C(=O)NCCOCCN(C(C(C)c2ccco2)=O)C)cnc(-c2cccs2)s1 N1(C(C2CCC(C)O2)=O)CC2(C1)CN(C(=O)CC1=CCCC1)C2.c12cn(nn1)C2=O C12(CC(O)C1)C(=O)N2.c1(C(=O)NCC2CCN(CCF)C2)conc1C1CC1 CC1(C)CCC(NC(c2cn(-c3ccc(Br)cc3)nn2)=O)C(c2ccccc2)C1 CCCC(C(=O)NC(C)CN(C)C(c1nsnc1O)=O)S(N)(=O)=O CS(=O)(=O)c1cc(C(N2CCC(NC(C3CCSC3)=O)C23CC3)=O)cc(N)c1 C(=O)(CCCCCNC(c1coc2c1COC2)=O)N(CC(C)(C)C)C1CC1 O=C(CCC#Cc1ccccc1)NCC1COCC1NC(C1(CO)CC1)=O C(C)(CCC(=O)NC(C)C(CO)NC(=O)C(c1ccnn1C)C)SC C(C(=O)N(C)OCC#C)NC(CNC(C1CC(=O)CS1)=O)=O.NC c1(NC(=O)NC(CC(=O)OC)Cc2ccccc2)cc(N)c(Br)cc1C N1(C(CC2(OC)CCC2)=O)C2CCC1CN(C(C1CC3CC3C1)=O)C2 c1(CN(C(C)C(O)C(=O)O)CCO)ccc(C(F)(F)F)c(F)c1 C(=O)(C1CCCc2nnn(C)c21)NC1C(CNC(CS(CC)=O)=O)CCCC1 C1(C(N(C2CCC(NC(C3(CO)CCOC3)=O)CC2)C)=O)CCC(C)(C)O1 CCN(OC)C(=O)C(CC1CC1)NC(c1ccn(C)c1C)=O c1(OC)ccc(C(N2CCCC(O)(CNC(=O)Cn3ccc(C)n3)C2)=O)c(O)c1 c1(-c2occ(C(=O)OC)c2)cccc2[nH]c(-c3nccn3C3CCOC3)cc12 N1(C(C(=Cc2ccccn2)C)=O)CC2CCC1C2NC(=O)C1=CSCS1 CCCCC(CNC(=O)C=C(CC)CC)NC(=O)CC1(O)CCOC1 c1(NCC(N2CCN(CC)CC2)(C)C)ccc(Cl)c(C)c1Cl c1(C(N2CCC(CNC(c3cc(C)nc(O)c3)=O)C2)=O)cc(F)c(C#N)c(F)c1 c1(C(=O)NCC(C)N(C(CC2C(C(=O)OC)C2)=O)C)sc2ncccc2c1Cl C12(CNC(c3c(N)ccc(F)c3)=O)CCC(CN(C(=O)C3=C(Cl)CCOC3)C1)C2 N1(C(CCCOCCC)=O)CC(NC(c2cnn(C)c2O)=O)C(C)(C)C1 C12(CC)CC(C1)C(=O)NCCN(CC1CC1)C2=O.C1CCCC1CC.CC c1(CNC(C(=O)Nc2cccc(C3CCCN(C)C3)c2)=O)ccc(F)c(N)c1 Cc1cccc(Cl)c1CC(=O)N(C1CCC(NC(c2cc(Cl)cn2C)=O)CC1)C Cc1cnn(C(C)C(=O)NCC(C2CC2)NC(=O)CC(C2CC2)C2CC2)c1.CC(C)C c1(OC)cc(NC(c2ccc3c(cnn3-c3ccccc3)c2)=O)cc([N+](=O)[O-])c1 C1(CNC(C2C(C(C)(F)F)C2)=O)CCCC(NC(=O)CCc2csnn2)C1 N1(C(CCCOCC)=O)CCCC(NC(c2cn3ccsc3n2)=O)C1C N1(C(CCC#C)=O)CCN(C(C2CC3CC3C2)=O)CC1CS(C)(=O)=O c1(CC(=O)NC2(C(=O)Nc3c(C(=O)OC)ccnc3)CC2)cccc(Br)c1F Cc1nc(CCNC(=O)CC(C2CC2)NC(=O)C=CCCC(C)C)n[nH]1 c1(OC)ccc2cc(C(N3CC(NC(C4CC4F)=O)CC4(CCC4)C3)=O)[nH]c2n1 C1(O)(CNC(Cc2n(C(C)C)cnn2)=O)CCCN(C(C2C=CCS2)=O)CC1 C=C(Cl)CCC(=O)NC(CN(C)C(c1coc(-c2ccccn2)n1)=O)CC CC1COc2c(C(=O)NCC3CCN(C(=O)CC4(CO)CC4)CC3O)cccc21 C(=O)(CCCC(C)N(C)C)N1C(CN(C(CNS(CC)(=O)=O)=O)C)CCC1 Cc1cccc(C(O)C(N2CCC(NC(c3nccn3C)=O)C2)=O)c1 C(c1nc2ccccc2s1)=CC(N1CC(CNC(=O)C=CCF)C(F)(F)C1)=O N1(CC(CC)CC)CCCC(C(=O)NC2CSC(C)C2)C1 Cc1cc(F)c(C(=O)NC(CO)CCCNC(c2ccn(C(F)F)n2)=O)cc1F c1(C(N(C)CC2CC3CC3N2C(=O)C(O)C(C)(C)C)=O)c(F)cc(Cl)cc1F CCC(C)(C)C(O)C(=O)NCC(C)NC(c1coc2c1CCCC2)=O c1(C(=O)NCC(CC)(C)NC(c2cc[nH]c2)=O)cc2c(Cl)c(OC)ccc2[nH]1 C1(C)(CNC(c2c(C)n[nH]c2)=O)CN(C(C2CCOC2=O)=O)C(C)(C)C1 C(=O)(CCCCCCN=[N+]=[N-])N1C(CNC(C(N(C)C)C2CC2)=O)CCCCC1 NS(=O)(=O)C(C(=O)NCC=CCNC(C1(CO)CCC1)=O)c1ccccc1 N1(C(C2(C)CN(N3CCCCCC3)C2)=O)CCCC(N=[N+]=[N-])CC1 N1(C(C)=O)CCN(C(=O)C(CC(F)F)NC(C23CCCC2C3)=O)CC1CCO N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(c2[nH]nnc2CC)=O)C1 c1(OC(C)C)cccc(OCC)c1.c12c(C)coc1NC(=O)C2.Cc1cnc(S)s1 C1(C(C(=O)NC(C2CCCC2)CNC(CN(C)CC2CCCC2)=O)F)CCCCC1 C=C(Cl)C(C)(C)C(=O)N1CC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2C(CCCN2C(=O)C(C)S(C)(=O)=O)C1 c1(C(=O)NC(C2CCN(C(c3c(CC)oc(C)c3)=O)C2)C)cnn2cccnc12 c1(CC(=O)NC2C(CNC(CC(=C)C)=O)CC2)c(F)cccc1Br c1(C(=O)NC(CC)CN(C(=O)C(C)OCCOCCO)C)cnc(C(C)(C)C)o1 c1(C(N2CC3(CC(NC(C4CCCCS4)=O)C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1O C(C(C)(C)C(C)(F)F)NC(C1(COC)CN(C(c2cc(C)c(F)cn2)=O)C1)=O Cc1nn(C)c(C(=O)N(C)CCNC(C2CC2c2ccc(Br)cc2)=O)c1Cl C=CCC(C)(C)CNC(=O)C(C1CCN(C(C2(SC(C)C)CC2)=O)C1)F C1(NC(c2cnnc(O)c2)=O)CCN(C(c2[nH]nnc2C(F)F)=O)CC1CO c1(C(C)C(=O)NC2(C)CC(NC(C3CCC3)=O)C2)ccc(-c2ccccc2)cc1 N1(C(CCc2n(C)cnn2)=O)CCCC12CCN(C(=O)COC1CCOCC1)C2 c1(C(N2C3CC(CNC(C=CC=CC)=O)C2CC3)=O)cc2nccc(Cl)c2s1 c1(N(C(C)C)C)nc(=NCc2ncn(C)c2Br)nc(N(C2CSC2)C)[nH]1 N1(C(C(CC)OC)=O)CC2CCOC2(CNC(=O)CCOC(F)(F)F)C1 N1(C(c2c(C)noc2C)=O)CC(NC(=O)C(C)OCC2CC2)CC12CCCC2 C1(NC(c2cc(C)c(C)[nH]2)=O)COCCN(C(C2CC23CC(O)C3)=O)C1 c1(C(=O)NC(C)CCNC(=O)CC2(C)OCCO2)cnc(O)c(C2CCCO2)c1 C1(CNC(=O)C=Cc2cn[nH]c2)CC2CCC1N2C(=O)CCc1cccc(Cl)c1 C1(CN2C(C(=O)NC3CC3)CNCC2)CCCCNC1=O C#CCCCC(=O)N(C)CC1CCCN1C(C1C2CCC(=O)C12)=O Cc1c(CNC2CCCCC2)cnn1CCO.c1(C2(C)CN2)nnnn1C(C)C c1(C(N2CC=CC(NC(CCc3c(C)n[nH]c3C)=O)C2)=O)ccc2nccn2n1 c1(C(N2CC(C(C)NC(CCNS(CC)(=O)=O)=O)C2)=O)ccc(C2CC2)nc1 N1(C(C)C)CCC(C(=O)NC2CN(C(C3CC4CC4C3)=O)CC2O)CC1 c1(CC(=O)NC2C3CCC2N(C(=O)C2=CCC2)C3)ccc2nc(O)[nH]c2c1 CN1C2CCC1CC(=CC(=O)NC(C)(CNC(C1CC(F)C(=O)N1)=O)C1CC1)C2 N1(C(C(c2ccc(O)cc2)OC)=O)CC(c2ccon2)(NCc2n[nH]c(=N)s2)C1 CC(C)C(O)CCN=c1[nH]c(=NCc2ccnc(OCCO)c2)c2ncccc2[nH]1 c1(CCC(N2CC(n3cc(-c4c(C)ocn4)nn3)C2)=O)ccc(Br)cc1 c1(C(=O)NC(CC(C)NC(Cc2c(C)n(C)nc2)=O)C)n[nH]c2c1CCSC2 Cc1ccc(CCC(=O)N(C)C)cc1C.C12C=CCN1C2 C1(C(=O)NCC2(CO)C(C=C)C2)CCN(C(c2c[nH]c(=NC)s2)=O)C12CC2 C(=O)(C1=CCCN(C(=O)CC=CCNC(c2cnc(C(C)C)o2)=O)C1)OC c1(C2C(C(=O)NC(CNC(CCC3CC(OC)C3)=O)C3CC3)C2)ccccc1Cl C1(NC(C2(NC(c3c(OCC)scc3)=O)CC2)=O)CC(C)OC1=O N1(C(=O)Cc2cncc(-c3cncc(C4CC4)c3)n2)CC(F)(F)OC(F)(F)C1 C1(C(=O)NC2C(NC(C3(OC)CC3)=O)C2)CC(C(C)C)C1 c1(CCC)nc(C(=O)NCC(C2CCCCC2)NC(=O)COCC(F)F)cs1 C1(=O)C(C(C)(C)C)C(=O)NCC(C)(C)CO1.N1(c2nnn(CC)n2)CCC(F)(F)C1 C1(C(=O)NCC(C2CCCCC2)NC(c2ccc(C(C)C)s2)=O)CC=CCC1C CCCC(CNC(c1cc(F)ccc1O)=O)C(=O)NC(C)CCSC N(C1CCCn2ccnc21)C(C1N(C(c2cc(C)no2)=O)CC1C1CC1)=O N1(C(CC(=O)NCC#C)=O)CC=C(CNC(C2CNC(=O)N2C)=O)CC1 Cc1oc(C(C)C)nc1C(=O)NCC1CCCCN1C(C1(C)CCC(=O)N1)=O c1(C(N2CC3C(CCNC(CC=C)=O)(CC3)C2)=O)nc2ccccc2cc1Cl C(C1CCCN1C(C1CC(F)CN1C)=O)=CC(=O)N(CC=C)CCOC O=C(C(O)CC(F)F)NC1(CO)CCN(C(c2cc(OC(F)F)ncn2)=O)C1 C1(N(C(c2cncnc2)=O)CC)CCCN(C(=O)C(C2CC2)C2CC2)C1 C1(O)(CC#C)CC(C(=O)N(CC(C)CC)C(C)C(=O)O)C1.N(C)CCC c1(C(=O)NC(CNC(C2C(C)OCC2)=O)(C)C)ccc(C#N)[nH]1 c1(C2(C(=O)OC)CC2NC(=O)C(F)(F)c2ccnn2C)ccc(F)cc1 Cc1cc(C)c(C(N2CCC3CN(C(=O)CC45CCC(CC4)C5)CC23)=O)c(C)c1 Cc1cc(C(=O)NC2CCN(C(C3CCC4(CCC4)O3)=O)C2C)cc(C)n1 CC1(C)CCC1C(=O)NCC1C=CCN1C(=O)COc1ccsn1 c1(CNC(c2cc(NC(C)=O)cn2C)=O)ccc(C#N)c(Cl)c1 C1(NC(CC2CCN(C)C2=O)=O)CCCN(C(c2nccc(Cl)c2F)=O)CC1 c1(C(C)(C)C(=O)NC2CCC(NC(=O)CCc3n[nH]c(=N)s3)C2)cccc(O)c1 c1(C(=O)NCC2(O)CN(C(C3CC(=O)N3)=O)C2)ncc(Br)cc1F C#Cc1ccc(C(=O)N(CC)CC2CCCN2C(=O)CC(CC)SCC)cc1 N1(CCC)CC(C(=O)N(CC(C)(C)NC(C23CCC2C3)=O)C)CC1=O c1(C(=O)NC2CCC(C)N(C(c3nccnc3N)=O)C2)c[nH]c2cc(Cl)ccc12 N1(C(CCSCC(C)C)=O)C2CCC1CC(CCNC(=O)C(F)n1cccn1)C2 c1(NC(C23CC(C(N4CC5CC4CO5)=O)(C2)C3)=O)ccc(Br)c(C(F)(F)F)n1 CN=c1ccc(C(=O)NCCC2(C(=O)Nc3cncc(C(N)=O)c3)CC2)c[nH]1 Cc1cccc(C(O)C(=O)NCCC2(CNC(C3CC(C)(C)O3)=O)CC2)c1F CC(C)C(O)C(C)C(=O)N1C2CCC(C(=O)NCC3CCC(C)C3)C1CC2 C1(NC(=O)C(O)C2CC2)Cc2ccccc2C1NC(=O)C1Cc2ccccc21 CCC(C)CC(=O)C(=O)NC1CCCC(NC(c2c[nH]cc2C2CC2)=O)C1 C1(NC(C2(NC(CC3CCN(C)C3)=O)CCCCC2)=O)CCC(=O)N(C)C1=O C(=O)(C(C)OC1CCCC1)N(C(C1CCCC1)CC)C C1(NC(C2C(C)=CCS2)=O)CCC(C)(CNC(=O)CN2CCN(C)CC2)CC1 c1(OCC(=O)NC(CCN(C(C)=O)C)C(C)C)ccc2c(c1)CCCC2=O C(C(C)C(F)(F)F)NC(=O)NCc1ncc(CC)s1 Cc1cn2cc(C(N3CCC(O)(CN(C)C(c4ccns4)=O)CC3)=O)sc2n1 C1(C(N2CCN(CCN(C(c3c(C)occ3)=O)C)CC2)=O)CCC2(C1)CC2(F)F c1(C(CCC)NC2CCC(CNC(=O)C(=O)NS(C)(=O)=O)CC2)cccc(Cl)c1 N1(C2CN(C(C3C(CC)CCC3)=O)C2)CCN(C(=O)CC23CCC(CC2)C3)CC1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)N1C2CCCN(C(C(=O)N(C)C)=O)C2CCC1 N1(C(C2CCN(c3ccc(C)cc3)C2=O)=O)CCN(C)CC12CCC2 c1(C(=O)OC)ccc(CN(C)C(=O)NCc2csc(-c3ncc[nH]3)n2)[nH]1 Cc1ccc(F)c(-c2cncnc2C(=O)Nc2cc(C#N)ccc2I)c1Br CCCC(C)(CCC)C(=O)NC(c1ccc(C)cc1)CNC(c1cocn1)=O NC1CCc2cccnc2N(C(c2cc(-c3ccccc3)co2)=O)C1 C1(C(=O)NC(CC=C)C2CC2)CC=CCN1C(=O)C1=NOCC1 c1(NC(=O)NC(c2ccccc2F)CCC)ccc(OC)c(OC)c1 C=CCCCCCC(=O)NCC(C(C)(C)C)NC(c1cc2sccc2n1C)=O N12CC(C(n3cccn3)C1)Cc1cn(nn1)CCC2=O.C1(SC(C2CC2)OC)CCC1 C=CCCCC(C(=O)NCCC1CCCCC1)NC(=O)CCNC(=O)COC c1(C(N2CC3(CCN(C(c4cccc(C)n4)=O)C3)C2)=O)cc2ccc(Cl)cc2o1 c1(C(=O)NCC2C3CN(C(C4(CC)CCCCO4)=O)CC32)cc2c(s1)CCOC2 C1(NC(C=CSC)=O)CC(NC(C2CC2c2cncn2C)=O)C(O)C1 C(=O)(C(CC1CC1)NC(c1ncoc1C)=O)NCC(C1CCC1)OC N1(C(CCN(C(c2c(NC)cccc2)=O)C)=O)CCC(C)C(CO)C1 C1(CNC(c2nnn(C)n2)=O)CCC(CNC(C2C3CCC(F)C23)=O)CC1 N1(C(c2c[nH]c(=N)s2)=O)CCC(CCCNC(=O)CC2CCCO2)CC1 Cn1cc(C(N)=O)c(C(=O)NCCOCCNC(C2CCO2)=O)n1 Cc1ocnc1C(N1CC(N(C(=O)CCN(C)C(=O)OC(C)(C)C)C)C1)=O C1(CCN(C)C(C2COCCN2CC(F)F)=O)CCN(C(=O)COCCO)CC1 CC1(C)CC(C(=O)N(CC(F)F)C2CC2)CN1C(C1CCC(CO)CC1)=O N1(C(c2c(C)coc2C)=O)CC2(CCN(C(C3C4CCCCCC34)=O)C2)C1 N1(C(C2N(C(c3c(CC)c[nH]c3)=O)CCC=C2)=O)CCC(CO)C1(C)C CN1CCOC(CCNC(=O)C(N2CCC(c3noc(C4CCCC4)n3)C2)=O)C1 C(=O)(CN=c1[nH]c2ccccc2s1)NCCN(C(C(COC)C)=O)C CC1CC(C(=O)N(C)Cc2ccccc2)CN(C(c2n[nH]cc2I)=O)C1 C(CCCCC(=O)N1CCN(C(c2n[nH]cc2C(C)C)=O)CC1)SC C(CCC(=O)N(CC(O)CN(c1ccon1)C)C)OCCO O=C1NCC2(CN(CNOC(=O)Cc3nccc4[nH]ccc34)C2)N1.C n1(C(C)C)cc(C(c2nnnn2C2CCCC2)NCc2cnn(C)c2)cn1 N1(C(CCC#C)=O)CCC(C2CCCN(C(=O)C(C)CC(N)=O)C2)CC1 CC(O)C(C)(C)CNC(=O)Nc1ccc(-c2cccnc2)cc1 c1(CCC(C)=O)cc(N2CCN(C(c3ccccc3)=O)CC2)nc(C(F)(F)F)n1 C(=O)(C(CC(F)F)N(C(=O)C=Cc1cnccn1)C)NCC(n1cccn1)C O=C(CCS(=O)(=O)c1ccc(F)cc1)OCc1cscc1C(F)(F)F C1(CNC(C(C)=C2CCCC2)=O)CC12CCN(C(c1ccoc1Cl)=O)CC2 C(C(CC(=O)Nc1cccnc1)C(F)F)NC(C(C)(C)N(C)C)=O C(=O)(C1Cc2c(Cl)cccc21)NCCNC(C1=C(CC)OCCC1)=O C(Cc1ccccc1)(CC(F)(F)F)N(c1nccc(Br)n1)C(C1CC(C)(C)C1)=O N1(C(c2nccc(C)c2)=O)CCC(C(=O)NC2(C3CCCCC3)CC2)CC1(C)C N1(C(c2ccc(COC)s2)=O)CC2CCC1C2NC(=O)CC1CCCC1O Cc1nc(NC2(CNC(C3CC(C)OC3C)=O)CC2)c(C)c(Cl)n1 C(C)(c1ccccc1OC)=CC(N1C2C(CNC(C(CC)(C)CO)=O)C(C2)C1)=O C=CCCC(C(=O)NCC(C)CC(=O)NC)NC(c1cnc2n1CCC2)=O c1(CCCC)sc(C(=O)NCCC2CCCN(C(=O)C=CCF)C2)cc1C N1(C(C=COCC)=O)CCC(C2CCN(C(c3cn(C4CCC4)nn3)=O)C2)C1 CCC(C)(CN=c1[nH]c(N2CCC=C(F)C2)nc(=N)[nH]1)C(C)O c1(C(N2CC3N(C(c4cccc(C)n4)=O)C3C2)=O)ccc2c(c1)n(C)c(=O)n2C C(C1=Cc2cc(Br)ccc2OC1)NC(C)(C)CS(C)(=O)=O C1(NC(C(n2c(C)ccn2)C)=O)CCCC(C(=O)NCCCN=[N+]=[N-])C1 O=C(CS(=O)(=O)CCO)NCC1CC(NC(C2OCCOC23CCC3)=O)C1 c1(OC)cc(OCC(C)OCC(C2CCOCC2)C)ccc1[N+](=O)[O-] CC1(C)CC(C(N2CC(OCCNC(C3CC=CCC3)=O)C2)=O)CNC1=O N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(C2CC2(C)C(C)C)=O)C(C)C1 C(CC(=O)NCC1(C(C)C)CC1)(C(F)(F)F)NC(CCC=CC)=O S(=O)(=O)(c1cnn2ccc(N(C)C)nc12)N1CCCC(CC)C1.C1CC(O)CN1 C1(CSC)CC2CCC1(NC(C1CC1c1ccnn1C)=O)C2.C1C(=O)NCCO1 C1(CCCNC(c2c(C(C)C)ncs2)=O)CCN(C(C2CCO2)=O)CC1 CN=c1[nH]cc(C(N2CCSCC2CCNC(=O)C#CC(=O)N(C)C)=O)o1 c1(-c2nc(C)c(NS(=O)(=O)c3ccc(Cl)s3)s2)c(C)ccc2ncccc12 c1(C(=O)NC2CCCN(C(CC=CCC)=O)C2)ccc2c(c1)oc1ccccc21 c1(C(N(C(C)CNC(=O)CC2C=CCC2)C)=O)ccn2c(O)nnc2c1 N1(C(C(F)=CCC)=O)CCN(CCCCCNC(c2cn(CC)nn2)=O)CC1 CCC(C)(O)C(=O)N(CC(=O)OC(C)(C)C)C.c1(CC)ccccc1Br C(=O)C(C)CS(C)(=O)=O.C(=O)(CS(=O)(=O)CC)OC(CC)CC N1(C(c2cnn(C)n2)=O)CCC2CC1CN(C(=O)CCn1cccn1)C2 C(=O)(C(CCS(C)=O)NC(N)=O)NCC1N(C(C2CCC(N(C)C)CC2)=O)CC1 c1(CNC2CCC(C(=O)Nc3cc(C)c(Cl)cn3)C2)c(O)cc(F)cc1F CCC(CC)(CN=c1[nH]c(C(C)(C)C)nc(=N)[nH]1)NC(c1cscn1)=O C1(CC(N2CC(n3cc(C4(C(C)C)CCC4)nn3)C2)=O)CC2CCC1O2 O=C1CCC(C(=O)NCC2CCCC2NC(=O)C(CO)c2ccccc2)=NN1 N12CC(O)CC1C2=O.C1(NC(=O)OCC)(CNC(=O)COC(F)F)CCC1 c1(N(C(=O)C(C)NC(c2ccc(OC(C)C)cc2)C)CC)ccc(Cl)cc1 N1(C(C2=C(C)CCC2)=O)CC2=C(C1)CN(C(=O)CC(C)n1ccnc1)C2 C(=O)(C1CCCc2sccc21)NC1CN(C(C2C(C)(Br)C2)=O)CC2(C1)CCC2 C(CC(N)=O)(C(=O)NCCOCCN(C)C(C1(F)CCCN(C)C1)=O)NC(C)=O c1(C(=O)NCC2C(NC(c3c(C)nn[nH]3)=O)C2)c(OC(F)F)cccc1Br C1(CC2C(OC)CCC2)CN(C(c2n[nH]cc2Br)=O)CC1=O S1(=O)(=O)c2ccc(Br)cc2N1C.N1(NCc2ccc(SC)o2)CCCCC1CO c1(OC)ccc(OCC(=O)NC2CCN(C(C3CC(O)CN3C)=O)C2)cc1 C#Cc1cc(C(=O)NC2CC(NC(=O)C(C)(CC)CC)C2)cc(N)c1 c1(C(N2CCC(NC(C=COCC)=O)C(C)C2)=O)ccc2oc(S)nc2c1 N1(C(C(CC#C)C)=O)CC(NC(=O)C(C)(C)CO)C(C2CC2)C1 C1(CCC)(C(=O)NC2CCC2CNC(C2CCC(O)CC2)=O)CCNC1=O C(=O)(C1COc2ccc(F)cc21)N1CC(NC(C2(CC#C)CCCC2)=O)C(O)C1 C1(CNC(c2ccn(C)n2)=O)CC2COCC2N1C(c1cc(Cl)on1)=O C1(C(C)C)CCCN(C(C2CC23CC(NC(=O)CNC(=O)C2CC2)C3)=O)CC1 Cc1cnn(C(C)C)c1C(=O)NC(C1CCOC1)COC(F)F C1(C(N2CC(n3cc(C(CN(CC)CC)C)nn3)C(C)C2)=O)CC(=O)NC(=O)N1 C(=O)(C(O)C(C)(C)CC)N1CCN(C(C2CCN(C(CC)=O)CC2)=O)C(CO)C1 N1(C(C(C)NS(CCC)(=O)=O)=O)CCC(N2CCN(C(C3CC3F)=O)CC2)CC1 N1(C(Cc2cn(C)nc2)=O)CCC(C2CCN(C(C3(CCF)CC3)=O)CC2)CC1 N1(CC)CC(COC(=O)Cc2csc(C(O)(C3CC3)Sc3ccccc3)n2)OC1=O N1(C(CCN(CCC)C)=O)CC(CC(=O)NCC2CCOC2(C)C)CC1C c1(C(c2nnnn2-c2ccccc2)NC(CSC)(C)C)cc(F)c(F)c(F)c1 c1(OC)ccc(NC(c2cnc(-c3cc[nH]c3)cn2)=O)cc1OCCO c1(-c2nc(CCCCCC)nn2Cc2ccsc2)ccc(F)cc1Cl c1(C(c2nnnn2Cc2cccs2)NC(c2cscn2)C)occc1Br c1(C(N(C2CCN(C(C(CC)(C)O)=O)CC2)C)=O)ccc(C(=O)OC)c(C)c1 N1(C(C23CC(C(=O)OCC)(C2)C3)=O)CCC(CNC(C2CCCC(C)O2)=O)CC1 Cc1ccc2c(C(N3CC4=C(C3)CN(C(C3CCOC3)=O)C4)=O)onc2c1 C1(N(C(CCC#C)=O)C)CN(C(c2cccc(OCC(F)(F)F)c2)=O)CC12CC2 N1(C(C(CNC(C2CCCC(O)C2)=O)N(C)C)=O)CCCCC(F)(F)C1 Cc1cc2c(=O)[nH]c(=O)n(CC3CCCC(F)(F)C(=O)N3C)c2n(CC=C)c1=O c1(C(=O)NCCN(C(=O)C(F)C2CCCC2)C)ccc(C#N)cc1.C12CC(C1)N2 Nc1c(C(=O)NCCN(C2CCCC2)C(C2CC3CC23)=O)cccc1F N1(C(c2n(CC)nnc2)=O)CCCC1(C)C(=O)NCC(C)(C)C1CCCC1 c1(OCC(=O)NCCCCn2cc(CCCS(C)=O)nn2)ccc(Cl)cc1Cl C12(C(=O)NCC34CC(CO)(C3)C4)CCC(CNC(C(CC)C(C)C)=O)(CC1)CO2 c1(NC(C2CN(Cc3ccncc3C#N)CCS2)C)nnc2n1CCCC2 Cc1scnc1C(=O)NCC1(C)CC1NC(c1ncoc1C(C)(C)C)=O CC(C)CC(C)(CO)NC(C1(C)CCCN(C(=O)COc2ccsc2)C1)=O Cc1oc(C(C)C)nc1C(N1CCCC(NC(=O)CCC2CCN(C)C2)C1)=O c1(C(=O)NCCN(C(c2cn(CCC)nc2C)=O)C)cnc(O)c2cccnc12 N1(C(c2cn(C)[nH]c2=N)=O)CCC(CO)(CNC(C2(Cl)CC23CCC3)=O)CC1 c1(OC)ccc(C(N2CCOC(C(C)Nc3cc(C(N)=O)ncn3)C2)=O)c(C)c1 C1(COC)(NC(=O)Cc2cccn2C)CN(C(=O)CCC2CCOC2)C1 C#CCCC(=O)NC(C1CC1C(=O)NC(c1nn[nH]n1)C1CC1)C N1(C(CN(S(C)(=O)=O)C)=O)CCCC(NC(C23CC(C)(C2)C3)=O)CC1 C1(NC(C2C(C=C)OCC2)=O)CCN(C(=O)CSc2c(C)n[nH]c2C)CC1CO C(=O)(C(O)CC1CCOCC1)NCC(CC)NC(=O)CCn1cc(Cl)cn1 c1(C(N2C(CCOC)CN(C(=O)C=C(C)Cl)CC2)=O)cnn2cc(C)cnc12 OCC(F)CN=c1[nH]c(=NCCc2ccsc2Br)[nH]c2c1CSC2 C1(NC(c2c(OC)ncc(Cl)c2)=O)CN(C(=O)CSC(C)C)C2(CCC2)C1 c1(C(=O)NC2(c3cn(CCN(C)C)nn3)CC2)cccc(C2CCOC2)c1 C(CC(O)C(=O)NCC(CC(C)C)NC(C1(C(=O)OC(C)(C)C)CCCC1)=O)SC c1(C(N(C(CNC(c2ccncc2F)=O)C2CC2)C)=O)ccc2ncccc2c1 N1(C(C)=O)CCN(Cc2ccc(Sc3ccccn3)c(F)c2)C(C2CCC2)C1 N1(C(CCn2ccc(C)n2)=O)CC2(C)CC1(C(=O)NCC(C)OCCO)C2 CC1CN(C(=O)C(C)(C)CN(C)C(c2cccc(C)c2N)=O)CCS1=O C1(CC(=O)NCCc2n[nH]cc2C(=O)NCC2(n3cnnn3)CC2)CCCCO1 c1(C(N(CC(N2CCCC2C(C)(C)O)=O)C(C)C)=O)nnc(S)n1C Cc1cc(C(N2CCC(O)(n3cc(C(=O)N(C)CCO)nn3)CC2)=O)cc(N)c1 N1(C(c2nc(C(C)C)oc2)=O)CC2CC1C2NC(=O)COc1ccsc1Cl c1(COC)ccc(-c2nc(-c3ccc(Br)cc3)nn2CC2CCCO2)cc1 CCC(C)(C(=O)NC1CC1NC(c1ccc(Oc2cccc(C)c2)cc1)=O)OC c1(C(=O)NCCC2(NC(C3C(C(C)(F)F)C3)=O)CCC2)ccc2nccn2c1 C(c1ccncn1)=CC(=O)NCC(CNC(C(c1ccccc1)OC)=O)(C)O C1(CC(=O)NC2C3CC2N(C(=O)COCC2CC2)C3)CCS(=O)(=O)C1 C=C(CNC(c1cnn(CCOC)c1)=O)CCNC(=O)CC1CCCC1C c1(NC(CN(C)C(c2cc(C(N)=O)no2)=O)(C)C)cc(O)ncn1 C12(NC(C(CC)CC)=O)CCCCCC1N(C(=O)C(C1CCC1)OC)CC2 c1(SCC(=O)NC2(CCCNC(C3(CCC)CC3)=O)CC2)ccc(O)cc1 Cc1nncn1NC(=O)C(C)N(C(=O)Cc1cccnc1F)C c1(C(N2C(C)CC(NC(=O)Cn3cnc(Br)c3)C2)=O)cc(F)c(N)cc1F C1(C(N(C2(CC(=O)NCCCCC#C)CC2)C)=O)CCCCC1O c1(SC)ccc(CCC(=O)NC(C)CC(C)NC(c2cnc(S)[nH]2)=O)cc1 c1(SC)ccc(C(=O)NC2CC2NC(c2n[nH]cc2C(F)(F)F)=O)s1 N1(C(C(CNC(=O)C#CC(C)(C)C)OC)=O)Cc2cccc(O)c2C1 CCCC(CC(C)C)C(=O)N1CCC(C(=O)N(C2CCCC2)C)C(C)C1 C1(NC(S2=C(CC)C(C)=C2)=O)CCN(C(C2CCN(C(=O)NC)C2)=O)C1(C)C c1(C(=O)N(c2ccccc2)Cc2cscn2)[nH]c2ccc(Br)cc2c1Cl c1(C(=O)NCCCNC(c2ccc(O)cc2F)=O)cc(F)c(Cl)c(Cl)c1 N1(C(C=CC(C)C)=O)CC(NC(c2ccc3nn(C)cc3c2)=O)CC12CCCC2 c1(NC23C(CNC(=O)OC(C)(C)C)CC(CC2)C3)ncnc2c1nnn2C(F)F C1(CC)CCc2[nH]nc(C(N3CCOC(CN(C)C(=O)C4CC4)C3)=O)c2C1 CN1C(=O)CCC1C(N1CC=CC1CNC(c1cc(C(N)=O)n(C)n1)=O)=O C1(C(N(CC(CC)C)C)=O)CCN(C(C2CCCOCC2)=O)CC1 c1(C(=O)NC(CNC(Cc2c(C)non2)=O)C2CC2)ccnc(C2CC2)c1 C1(OC)CN(C(=O)CC2CCCC2)C(C)(CNC(c2sccc2F)=O)C1 C1(CNC(CCSCC)=O)CCC(NC(C2CC2C(F)(F)F)=O)CC1 O=C(C1=CCCOCC1)NC12CCCC1N(C(c1cnns1)=O)CC2 O=C1CCN(C)C2CCCCCN12.c1(CC(=O)OC(F)F)ccc(F)c(I)c1 C1(OCC)CC(CC(=O)NC(C)CCNC(c2cnc[nH]2)=O)C1 c1(C(N2CC(C(C)(C)NC(=O)CC3COC(=O)C3)C2)=O)cc([N+](=O)[O-])ccc1N N1(C(c2ncc(CC)s2)=O)CCCC(O)(CNC(c2cn3ccnc3s2)=O)C1 c1(C)ccc([N+](=O)[O-])[nH]1.c1(C(=O)NC2C(NC(CNC=O)=O)CCC2)ccccc1O C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(c1cc(OC)no1)=O C(=O)(C1=NOC2COCC12)N1CC(C(=O)NCCC(C(F)(F)F)N(C)C)OCC1 C(=O)(C#CC1CCOC1)N1CCC(C(=O)Nc2cccc(F)c2)OCC1 C1(c2cn(C3CCCC3O)nn2)(N(C)C)CCN(C(=O)CCC2CCCCO2)C1 CC(CC(=O)N(C)Cc1ccsc1)C(C)(C)NC(C12CCC(CC1)C2)=O CC1CCC=C1C(=O)NCC1CSCN1C(=O)CCc1ccccc1 c1(C(=O)NC2CC(C)(CNC(C3(C(=O)NC)CC3)=O)C2)c[nH]c2c(Cl)cccc12 CCC(CCC(=O)N(C)CCNC(=O)C(C)CC(N)=O)NC(=O)OC(C)(C)C C1(C(C)C)CNC(=O)CN1C(=O)C(C)(C)C(C)NC(=O)C1=CCSC1 CC1=C(C)CN(C(=O)C(CNC(C2CC2(C)C(C)C)=O)N(C)C)CC1 c1(OC)ccc2c(n1)NC(C(N1CCCC1CN(C)C(C1(SC)CCC1)=O)=O)C2 CS(=O)(=O)c1ccc(C(=O)NNC(=O)Cc2ccccc2Br)cc1 C(=O)(C(O)(C(F)(F)F)C1CC1)N(CCCN(C(C(CCCC)N(C)C)=O)C)C Cc1nc(C2CC2)ncc1C(=O)NC1CCN(C(C2(C3CC3)CC2)=O)CC1O C1(CC(=O)NCCN(C(C2CCCCCC2)=O)CC)CCC(F)(F)CC1 C(=O)(CCCCC(=O)NC1CC(CO)N(C(=O)CCOCC(F)F)C1)NC c1(OC)cccc(Cl)c1C(N1CCN(CCN(C(=O)C(C)CC(C)C)C)CC1)=O c1(C(=O)NCC(CC=C)NC(c2c[nH]cc(C)c2=O)=O)c(F)ccc(C#N)c1F C1(NC(CCCN(C)C)=O)CC(NC(C2OCCC2C(F)(F)F)=O)C(O)C1 c1(C(N2CC(NC(c3c(CC)non3)=O)C(C)(C)C2)=O)nn(C)cc1[N+](=O)[O-] C(=O)(C(CCF)NC(=O)CCc1ccccc1)NC(C)CN=[N+]=[N-] N#Cc1ccc(=NCCC(=O)N2CCC3(CCCCC3NC(C3CSC3)=O)C2)[nH]c1 C1(N(C(C2(OC)CCSC2)=O)CC2CC2)CCN(C(=O)CCNC(N)=O)CC1 C1(NC(C2(C=C)CCOCC2)=O)CCN(C(=O)CC2CCCN(C)C2)CC(O)C1 CCCC(C(=O)NC1CCOC1C(N1CC=CC1)=O)C(C)C C1(OC)CC(NC(C2CCCC2)=O)CN(C(c2nn(C)c(Br)c2C)=O)C1 c1(CSC(C)(C)C)ccco1.C(CCCNC(n1cncn1)=O)N(C(=O)CSCC)C C(=O)(C(CCc1ccccc1)C(F)(F)F)OC(C)C(N1CC(C)(C)OC(C)(C)C1)=O C1(CNC(CCCOCC=C)=O)CCCN(C(=O)Cc2c(Cl)cnn2C)C1 CN1CCn2nc(C(c3nnnn3C3CCCCC3)NC3(COC)CC3)cc2C1 N1(C(C2C(NC(c3cnn[nH]3)=O)C3CCC2C3)=O)CCC(C2CCC2)C1 c1(C(N2CC3CC(NC(C4(Br)CC4)=O)CC3C2)=O)ccn2cncc2c1 Cc1cc(OCC(=O)NCC2CC(C)N(C(c3n[nH]cc3F)=O)C2)cc(C)c1 c1(C(=O)NCC2(CNC(c3ncn(CC)c3)=O)CC2)cccc(N2CC=CC2)c1 Cc1cc(C=CC(=O)NC2CN(C(=O)COC(=O)CO)CC2O)on1 N1(C(C(C)CSc2ccccc2)=O)CCCC(CO)(NC(=O)C2=CSCCO2)C1 C1(C)(CC)CC(NC(C2CC=CC(NC(=O)C(C)(C)CSC)C2)=O)CCO1 C1(N(C(C(CCC)N(C)C)=O)CC)CCCN(C(c2nn(C)cc2C)=O)CC1 c1(OC)ccc(C=CC(=O)NC(C)CN(C(=O)C(F)CC2CC2)C)c(OC)c1 c1(N2C(C)CC(F)C2)ccc(S(=O)(=O)NCC2CC23CC3(F)F)cc1Cl Cn1ncc(C(N2CC(NC(=O)CC3C=CCC3)CC(C)(C)C2)=O)c1S(C)(=O)=O C(=O)(C(F)(F)C(F)(F)F)NC(C(C)(C)NC(c1cc(C)[nH]c1C)=O)C CC(C(=O)N1CC2(CC(NC(=O)CC(C)NC(=O)OC(C)(C)C)C2)C1)C(C)(C)C c1(C(C(=O)NCC(CC)NC(c2cocn2)=O)(C)C)ccc(Cl)cc1 N1(C(CNS(C)(=O)=O)=O)CCC(C)(C)C(NC(C2(O)CCSCC2)=O)C1 c1(C(=O)NC2CCCC(NC(c3cc(C)c(C)[nH]3)=O)C2)cnc2nccn2c1 Cc1nn(C)cc1C(=O)NCc1csc(C(=O)NCC(c2ccccn2)C)c1 C(=O)(CC1=CCCC1)NCC1C(C)CCN1C(=O)CCOC1CC1 c1(C(N2CC(N(C(c3c(C)scn3)=O)C)C2)=O)ccc2c(Cl)ccnc2c1 C1(NC(Cc2cc(C)n(C)n2)=O)CCN(C(c2nnn(C)c2C)=O)C12CC2 C1(C(=O)NCc2ccc(NC(C)=O)cc2)CC12CCCCC2 C1(C(=O)NC(CC(=O)OC)C)CC12CCN(C(c1cc(OC)nc(C)c1)=O)CC2 C1(NC(=O)CC2CCOC2)CCN(C(=O)CNC(C2CCC2)=O)CC1CO N1(C(C2(NC(C)C)CC2)=O)CC2(CCN(C(C3(C)COC(=O)C3)=O)C2)C1 N1(CCC(CC)(C)C)CCC(=O)N(Cc2ccc(CC(C)C)cc2)C1=O CCCCN(C1(CC(=O)OC(C)(C)C)CC1)C N1(C(C(C2CC2)NC(=O)CC2COCCOC2)=O)CCn2ccnc2C1 C#CC1CCN(C(=O)C(CC)N(C)C(c2coc(N(C)C)n2)=O)CC1 c1(C(N2CC3N(C(Cc4c(C)ccnc4)=O)C3C2)=O)c(F)ccc(F)c1Cl S(=O)(=O)(c1ccccc1[N+](=O)[O-])NC1CN(C(C2CCCC23CC3)=O)C1.CN1CC1 c1(N2CCN(c3ccnc(C(C)C)n3)CC2)ccc2c3c(cccc13)CC2 C#Cc1ccc(C(=O)NCC2CC2CNC(=O)Cn2cc(Br)c(C)n2)c(C)c1 CCC(C)C(=O)C(=O)NCC1CC2(CC(NC(=O)CC3CC=CCC3)C2)C1 N1(C(C2(CC)CCC2)=O)C(C(=O)NCCOCC2CCC2)CCC12CC2 C1(NC(C23CC(NC(C(CC)OC)=O)(C2)C3)=O)CCCC(C(C)C)C1 N(C(=NCCCCl)N1CCC(n2cc3ccccc3n2)C1)CC1C(C=C)C1 N1(C(CCC)=O)CCCCC1C(N1CCC(N(C(c2ccncc2)=O)CC)C1)=O C(=O)(CC1OCc2ccccc21)N1CC(C(N)=O)(CNC(CC(C)O)=O)C1 N1(CC(=O)NCCC(C)NC(=O)C(F)=CCCF)CC(=O)Nc2ccccc21 N1(C(C2CCCC23CCC3)=O)CC(C2CC2)(C(N2CCOC3CC23)=O)C1 C1(C(=O)OCC)CCCCC1NCc1cc(C(F)(F)C(F)(F)F)on1 c1(C(=O)NCC(CC(C)C)NC(C2(OCC)CC2)=O)c(O)nnc(C)c1C C(=O)(C1=CCCCC1)N1CCC(=CCNC(CN(C)C(c2ccccc2)=O)=O)CC1 C1(CCC(=O)N(CCNC(C(C)CO)=O)C)CCC(O)CC1 CC1CCC(CO)(NC(=O)CCN(C)C(c2cccc(CC#N)c2)=O)C1 N1(C(C(CC(N)=O)O)=O)CCOC2CN(C(C3CCCO3)=O)CC12 C1(C(=O)NCC(C2CCCC2)C)Cc2c(F)cccc2C(=O)O1 Cc1oc(C(N2CCC(CN(C)C(C3(C(C)C)COC3)=O)C2)=O)cc1Br Cc1cc(C#N)nc(N(C2CCN(C(c3cnc(O)n3C)=O)C2)C)n1 N1(c2cc(NCC(c3ccccc3Cl)N(C)C)ncn2)CC2CC(C1)C2CO c1(-c2n(CC(CC)(C)CO)c(N(C3CCCCC3)C)nn2)ccc(C)c(F)c1 CC1=C(C(=O)N2CCC(CNC(=O)CCN(c3cnccn3)C)C2(C)C)CCO1 N1(C(c2cc(CC)[nH]n2)=O)CCC2CN(C(C3CC4(CCC4O)C3)=O)C2C1 c1(CC(=O)NCC2C(NC(c3cc(C)oc3)=O)CCCC2)cc(F)c(C)cc1F N1(C(C2(CC)CCCC2)=O)CC(N(C(=O)C(n2cc(C)cn2)C)C)C(O)C1 C1(CC=C)(C(=O)NCC(=O)OC)CCN(C(=O)CCCOCCC)C1 c1(CC)nn(C)c(C(N2CCC2CNC(=O)CC2CCC3(CCC3)O2)=O)c1Cl N1(C(C(=O)NCCOCC)C(C2CC2)OC)CCC2OCCCC2C1 N1(C(C(C)n2cccn2)=O)CCC2(NC(=O)CCc3ccc(O)nc3)CCCC12 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(C(C2C(C)(C)C2(F)F)=O)C1)F C1(NC(CC(C)CF)=O)CCC2(CC1)CC2NC(=O)CCN1CCC(O)CC1 c1(C(=O)NC2CN(C(c3nnc(C)s3)=O)C2)ccc(=O)n2c1CCCCC2 N1(C(C2C(NC(c3cc4n(n3)CCO4)=O)CCC2)=O)CC(=O)N2CCCC2C1 c1(N2CCC(NC(c3cc(CCC)oc3C)=O)C2)ncc2c(n1)COC2 c1(C(N2C(C(C)NC(C=C3CCC(C)CC3)=O)CCC2)=O)cnn2cccnc12 c1(CNC(C2(c3cccc(OC)c3)CC2)=O)c(Cl)ccnc1F Cc1oc(C(=O)NC(CCN(C)C)C(=O)NC2CCN(CCCO)C2)cc1CO CCS(=O)(=O)CC(=O)NC1CCCC1(C)CN(C)C(c1ncnc(C)c1C)=O C(=O)(C(C)CS(C)(=O)=O)N1CC2(N(C(C(CCC)CC=C)=O)CC2)C1 C1(C(=O)NCCN(C(=O)CC2CCCC(C#N)C2)C(C)C)CC2CCC1C21CC1 Cc1cc(C2CC2)ccc1C(N1CCC(C)(CNC(c2cnncc2O)=O)C1)=O N1(N(C(C(C2CCN(C(CN3CCC(C)C3)=O)C2)C)=O)C)CCC(C#N)C1 C1(CN(C(c2c(CC)occ2)=O)C)C2CN(C(=O)Cc3csc(C)n3)CC12 C12(C(=O)Nc3cc(SC)n[nH]3)CC1CN(C(c1nc(Br)cs1)=O)C2 Cc1c(Cl)ccnc1C(=O)NCCN(C(c1csc(O)n1)=O)C(C)C C1(C(=O)NCc2c(C)noc2C)CC(O)C(O)CO1 C(CCC(=O)NC(C)CNC(=O)C(C)(C)C1CC1)NC(=O)OC CC1CN2CCCC2CN1C(c1csc(S(N)(=O)=O)c1)C(=O)NC1COC1 C1(OC(C(c2c(C)n[nH]c2C)C)=O)CC2CCC1CC2 N1(C(C2C(OC)CCC2)=O)CCC(N=[N+]=[N-])(C(=O)NC2CCCCC2CCO)C1 c1(C(=O)NCC2(OC)CN(C(C3CCC(F)C3)=O)C2)cnn2c1CCC2 C1(OC)CCCC1CNC(=O)C(C1CC=CCC1)NC(=O)Cc1nocc1C c1(C(=O)NC(C)CN(C)C(C2CCCCS2)=O)ccnc(C2CCC2)c1 c1(C(=O)NC2(C3CCCN3C(=O)CCn3cccc3)CC2)cc2n(n1)CC(F)C2 N1(C(C(C2CCC2)OC)=O)CCN(C(=O)CCc2conc2C)CCC1C c1(C(N2CC(NC(C(C=C)c3ccccc3)=O)C2)=O)c(C)cc(C)oc1=O Cc1cccc2ccc(C(=O)NC3CCC(NC(=O)C(C)O)C3)nc12 Cc1cccc(N)c1C(=O)NC1CCCC(NC(=O)C=CBr)CC1 CCCCC(CCC)NC(=O)C=CC(C)(C)NC(c1cc(C2CC2)[nH]n1)=O C1(CNC(C(CSC)(C)C)=O)CN(C(=O)CCCC#N)CCC1C c1(NC(C2CC3(CC3)CN2C(C2CC=CCC2)=O)=O)cc(Br)cc2[nH]ncc12 Cc1cnc(C(=O)N(C)CC2(NC(=O)CC3CCCCCCC3)CC2)cc1Cl c1(OC)ccc(C=CC(=O)NC2CC(F)(CNC(=O)CCCC3CC3)C2)c(C)c1 c1(C(C)C)ccc(C(C(C)C)NCc2cncc(-n3ccnc3)n2)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C2C(CNC(C(C(C)C)O)=O)CC(CC2)C1 c1(C(=O)NCCSc2cccnc2)cnc2ncnn2c1O N1(C(Cc2c(C)cccc2C)=O)CCC2CN(C(c3ccnnc3O)=O)C2C1 N1(C(C(CC=C)C)=O)CCN(C(c2cc(C)c(C)o2)=O)C(CCO)C1 C1(C(=O)NC2CC(NC(CCCOCCC)=O)C2)CCC(=O)N(C(C)C)C1 c1(NCC2(C)CCCN(C(CC(CN(C)C)O)=O)C2)ncc2c(n1)CCCCC2 C1(NC(C2CC3CC3C2)=O)CCCCCN(C(=O)C(F)(F)C2CC2)C1 Cc1cc(-c2nn[nH]n2)cc(N2CCCC(C(=O)N(C(C)C(N)=O)C(C)C)C2)n1 C=CCC(CC)C(=O)NCCCOCCNC(=O)CC1CCC(C)(C)CC1 C12(C(N3C4CCC(NC(C5C(C)C5)=O)C(C4)C3)=O)CCC(C#N)(CC1)CC2 CC(C)C(C(C)C)NC(C1CC(NC(=O)COCCN(C)C)CCO1)=O c1(C(N(CCNC(C(C2CCC(=O)N2)C)=O)C)=O)cc(=O)n(C)o1 c1(C(=O)NC(C(C)NC(c2ccc(C(C)=O)[nH]2)=O)C)ccc(C(F)F)nc1O C(=O)(CC(O)C(C)(C)C)N1CCN(C(C(C(C)C)NC(=O)OC(C)(C)C)=O)CC1C C=CC(CCC)CC(=O)NCc1cc(C(=O)NC(C)C(C)CO)on1 C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)N1CC(NC(c2c(CC)cno2)=O)C(C)C1 N1(C(C(CC)=CC)=O)CCN(C(C2COCCN2C=O)=O)C2CS(=O)(=O)CC12 c1(N(C2C(CNC(CC3(OC)CC3)=O)C2)C(c2c[nH]c(=N)s2)=O)cccc(Br)c1 C12(NC(C(N3CCN(C)CC3)C)=O)CC(CNC(C3CC(C#N)C3)=O)(C1)OC2C c1(CC)ccc(OC)cc1NC(=O)C(c1ccccc1)SC.C1(C)CO1 N1(C(CC=CC)=O)CC(OC)CC1(C)CNC(c1cocn1)=O C1(C(=O)NCC(CC)NC(c2cc(C)n(-c3ccc(C)cc3)n2)=O)CCCN(C)C1 c1(CC)sc(C(=O)NC(C)CCNC(=O)C(C)OCC(C)C)cc1C Cc1cccc(OCCC(=O)NCC2C3CN(CC4CCC(C)O4)CC23)c1C c1(SCC(=O)N(C(CNC(=O)CCn2cccc2)C2CC2)C)ccncc1 C=CC(CC)CC(=O)NC1CN(c2cc(C(F)(F)F)nc(C)n2)CCC1C Cc1cc(C(=O)NCC2CCCCC2C(=O)NC(c2cc[nH]n2)C)cc(C#N)c1 CCCCC(CNC(=O)CCc1nccn1C)NC(c1ccc(C(C)C)s1)=O N1(C(C(C)OCC2CC2)=O)CC(C(C)(C)O)(NC(C2CC2(C)Br)=O)C1 CCC(C)(C)C(C)NC(=O)C(C)(C1CC1)N(C(=O)Cn1ccnc1)C c1(C(=O)NCC2(CN(C(C(CSC)O)=O)C)CC2)cc2c(F)ccc(F)c2[nH]1 C(=O)(CC1=CCCCC1)NCCC(=C)CNC(=O)C(F)(F)c1ccnn1C C12(CNC(c3ccnnc3)=O)CCCN(C(=O)Cc3cccc(F)c3F)C1C2 N1(C(c2cnc(CC)[nH]2)=O)CCC(C)C(NC(c2cn3cnnc3cn2)=O)C1C C1(C(=O)NCCC(=C)C)COCCC1NC(c1ccn(CCOC)n1)=O S(=O)(=O)(c1ccc(NCCCOC(C)(C)C)c(F)c1)N(C1C(C)OC(C)C1)C N1(c2n(CC)c(CO)nn2)C(C)CCCC1C.C(=O)(CCN=[N+]=[N-])N C#CCCCCCCC(=O)N1CCCC(C)(NC(=O)C(C2CC2)OC)CC1 C=CCC(F)(F)C(=O)N1CC(CCNC(=O)C(C)NC(C2CCCC2)=O)C1 N1(C(C(C(C)C)OC)=O)CC2CCC(C1)C(NC(=O)C(c1cccnc1)O)C2 C1(NC(=O)OC(C)(C)C)CC2(C1)CC(CC1CN(c3nccnc3C#N)C1)C2 CC(C)CCCCCC(=O)N1CCC(C)C1C(=O)NCC1OCCC1(C)C C1(C)(CNC(C2(OC)CC(C)C2)=O)CN(C(c2cnc(C)c(N)c2)=O)CCO1 C1(C(=O)Nc2cnc(C(F)(F)F)nc2)CC2CCC1N(C(C1CCCC1)=O)C2 C=CC(C)(C)CC(=O)NC(C)CCN(C(=O)C(F)C1CCCC1)C O=C(CC1=CCCCC1)NCC1CCCC(NC(=O)CCCn2ccnc2)C1 C1(CNC(c2cnn(-c3nccs3)c2)=O)CC(F)CN1C(=O)CO CN1CCC(C(N2CCCC(C(F)F)C2)=O)(NC(c2cccnn2)=O)C1 C1(NSc2nnnn2Cc2ccc(-c3ccc(C)cc3)o2)CC2(CCCOC2)C1 N1(C(C(COC)OC)=O)CC=CC(NC(C2(CC3CC3)CCC2)=O)C1 N1(Cc2c(CSc3ccc(Cl)cc3)cccc2)CCOC2(CCCC2)C1 C1(CC(N2CC(CNC(c3c(C)nc(N(C)C)s3)=O)C2)=O)CCCCCCC1 c1(CCN(C2CCN(C(=O)CC3COCCO3)C2)C)c[nH]c2ccccc12 Cc1cncc2nc(CC(=O)NCC3(C4=CCNCC4)CC3)cn12 CC1(C)CCC1C(=O)NCC1(NC(C2(c3ccccc3)CC2)=O)CCC1 CN=c1ccc(Br)c(C(=O)NC(C)CN(C(=O)CCC(C)C)CC)[nH]1 c1(CCNC(NCC(=C)Cl)=NCCCF)c(N2CCOCC2)cccc1CC C(=O)(CC(CNC(=O)CC1CCCN1C)NC)NCC1(CCC)CC1 N1(C(CCn2c(C)cc(C)n2)=O)CCN(C(C2CC23CC3)=O)CC1C(C)(C)C C1(NC(C2(F)CC(C(=O)OCC)C2)=O)CC(NC(=O)C2=NOCC2)C(O)C1 C=CCC(CC)C(=O)N1C(CC(N2CC(C)CCC2CC)=O)C2CCCC12 Cc1ccc2nc(CNn3cccc(N)c3=O)ccc2c1 C1(C(N2CC(CNC(=O)Cc3ccno3)C2)=O)CC12C(=O)Nc1ccccc12 C(=O)(C(CO)C(F)(F)F)NCCC(=O)NCc1nccc(OC)n1 C(=O)(CC(c1ccccc1)NC(N)=O)NC(c1ccc(-c2nn[nH]n2)o1)C C(=O)(C(C(=O)OCC)C(C)C)NC1(F)CN(C(C(=O)NCCN(CC)CC)=O)C1.CSC C1(NC(C(C=CC)O)=O)CCN(C)C12CCCN(C(C1CCC(C)C(C)C1)=O)C2 C(CC(C)(C)C(=O)N1CCCOC(CNC(C2NC(=O)OC2(C)C)=O)C1)OC c1(C(=O)NC2(CNC(=O)Cc3c[nH]ccc3=O)CC2)cc2c(Br)cccc2[nH]1 C1(NC(CC2CCC(=O)N2)=O)CCOC12CCN(C(=O)C#CC1CCC1)CC2 C(C1=CCN(C(C2(C)CC2Br)=O)CC1)NC(C(CC)Oc1ccccc1)=O C(CCCC(=O)N1CCC1C(C)O)N(C(C(C)(C)OC(C)=O)=O)C C1(C(N(C(C)C)CCN(C)C(C2CCC(F)C2)=O)=O)CCn2ncnc2C1 C1(C(=O)NCCCCCNC(c2cnc(C(C)(C)C)[nH]2)=O)(COC)CC=CCC1 N1(C(c2ccc(C(C)O)cc2)=O)CCC12CN(C(=O)CN1CCC(F)(F)C1)C2 C1(NC(Cc2c(C)non2)=O)CCCC(NC(c2c(Br)noc2C2CC2)=O)C1 C1(C#CC(=O)NC2COCCN(C(=O)CC(C)C3CC3)C2)(CC)COC1 c1(C(N2C(CCNC(Cc3cc(C)no3)=O)CSCC2)=O)csc2ccccc12 C1(C2CCOCC2)(C(N(C)CCN(C(=O)C(C)(C)C(N)=O)C)=O)CCOCC1 CC1CCCC(C(C2CC(C(C)C)C2)=O)(CNC(C23CCC(NC)(CC2)C3)=O)C1 C1(CC)CCCN(C(=O)C(C)SC)C1C(=O)NC1CC1C(=O)NCCO Cc1cccc(C(=O)NC(C2CN(C(c3cc(Cl)ccn3)=O)C2)C)c1[N+](=O)[O-] C1(NC(C(COC)(C)C)=O)CC12CCN(C(C1CC(CF)C1)=O)CC2 N1(C(=O)Oc2ccccc2)CCS(=O)(=O)N2CCOCC12 CC1(C(=O)NC2CC(NC(=O)CCC#N)CC2O)CCC2(CC1)CC2 C12(C(=O)Nc3nc4ccc(C)cc4s3)CC(C(=O)NCC#N)(C1)OC21CCC1 c1(CNC2C(C(=O)Nc3nc(C)c(Cl)s3)C2)ccc2cc[nH]c2c1 CCCCCCCCCCNC(=O)CS(=O)(=O)Cc1c(Cl)cc(C(F)(F)F)cc1Br C1(CC(=O)N(CCOCC=C)C)COCCN1C(=O)CC1(O)CCCOC1 C1(O)(CCC)CCN(C(c2c[nH]nc2CNC(=O)C(C)NC(C)=O)=O)CC1 N1(CC(C)C)N=C(C(=O)N(CC(C)O)CCNC(=O)CCCS(C)(=O)=O)CCC1=O Cc1nc(C(=O)N(C)CCc2ccccn2)c(=O)[nH]c1C C1(OCC(N)=O)CCN(C(=NCC2(CO)CCCCC2)NCC)C1.C1(N)CCC1 c1(C(N2CCC(NC(C(C)SCCCC)=O)C2)=O)cccc(C)c1[N+](=O)[O-] N1(C(C2(COC)CC2)=O)CC2CCC1C(CNC(=O)C(O)CC(C)C)C2 C(=O)(CCCCOC)N(CC(=O)NCCn1cnc(CO)n1)CC c1(SC)cc(C(=O)NCC2CN(C(=O)CCC3CC3(C)C)CCO2)c(C)o1 N=c1nnn(CC(=O)NCC2CC2NC(c2cn(CC(F)(F)F)nn2)=O)[nH]1 CC12CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CN(C(C1CNC(=O)N1)=O)C2 C1(CC(=O)Nc2cccc(F)c2)CN(C(C2CC=CCC2)=O)CCO1 c1(C(=O)NC2CC(N(C(CC(c3ccc(F)cc3)C)=O)C)C2)c[nH]ccc1=O CCC(CC(=O)NCC(c1ccccc1F)NC(=O)C(C)(C)COC)CC(C)C c1(C(=O)NC2CCCN(c3nnc(C)o3)C2)ccc(O)nc1C N1(C(C23C(CN(C(C)=O)C2)C3)=O)C2CCC1CC(NC(C1(C)CS(=O)(=O)C1)=O)C2 C(c1ccc(F)cc1)=CC(=O)NC1CC(CNC(C(COC)C)=O)C(O)C1 N#Cc1cc(NCC(O)CNC(=O)Cc2csc(Cl)c2)nc(C(F)(F)F)n1 Cc1ccc(C(C)C(=O)NC(C)(C)CNC(c2sccc2F)=O)s1 Nc1ccc([N+](=O)[O-])cc1C(N1CCC(NC(=O)CC2CCOC2)C1)=O C1(NC(=O)C=C2CCOCC2)CCCN(c2nccn2C)C1.CC1CNC(=O)N1 CC(C)CC(CC(C)C)C(=O)N(C)CC1(NC(=O)CN2CC(C)(C)C2)CC1 Cc1ccnc(CNC(C2CC3CC3N2C(=O)CC2CCOC2)=O)n1 C1(C(=O)NC2CC(OC)(OC)C2)CCCC(N)C1.N(C)(S(N)(=O)=O)CC(=O)NC1CC1 c1(CNc2nc(C)nc(N3C(C)CC4CNCC34)c2)ccc2ncccc2c1 C(CN=c1[nH]cnc2ccccc12)Sc1c(C#N)nccc1 c1(C(=O)NCC2(NC(C=C(C)C(C)C)=O)CCOC2)cc(C)cc2c1CCC2 Cn1ncc(C(=O)NC2CC(F)(CNC(c3ccc(CO)cn3)=O)C2)c1F C(=O)(CS(=O)(=O)C1CC1)N1CC(CNC(c2cc(F)cnc2O)=O)C(O)C1 c1(C2C(C(N(C(C(=O)N3CC(COCC)C3)C3CCC3)C)=O)C2)ccccc1F N1(C(C(c2ccccc2F)OC)=O)CC(F)(F)CC1CNC(c1ccccc1C)=O C(CCCC(C)NC(=O)CC(C)C)NC(C(C)OCCCC)=O C#Cc1ccc(F)cc1NC.c1(CN2CC(CO)NC2=O)ccccc1 C(CCC(=O)N1CC(O)(CNC(=O)CC2CCOC2)C1)SC n1(CC(=O)NCC(CCNC(CC(C)CN(C)C)=O)O)sc(=O)c2ccccc12 c1(C(N(CCCNC(c2c[nH]cc2-c2cnn(C)c2)=O)C)=O)ccc(N)cn1 Cc1ncc2n1CC(C(=O)NC(C)CC1(O)CCC1)CC2 C1(C(N2CCC(CN(C(=O)CC(C)NC(N)=O)CC)CC2)=O)CCC(=O)N(C)C1 c1(C(=O)NC23CC(NC(CC4CCC(C)C4)=O)(C2)C3)ccc2c(c1)OCO2 N1(C(CSCC)=O)CCC(O)C1.C(=O)(CCCN(C)C(C)=O)N(CC#C)C C1(C(N(CCC)C)=O)CCCCC1OC.C1(O)(C)CN(C(=O)CCCn2cccn2)C1 N1(Cc2c(C)scn2)CC2C(C(=O)Nc3n[nH]c(C)c3Cl)C2C1 c1(CC(=O)NCCCNC(=O)Cc2cn[nH]c2)c(F)cccc1F c1(CN2CCC(C(=O)Nc3cccc(CO)c3)C2)ccc(-n2ccnc2)cc1F c1(C(N(C)CCC2CCN(C(c3cnc(Cl)cn3)=O)CC2)=O)cnc(O)nc1O Cc1cc(Br)c2nc(C(N3C4CCC3CN(S(=O)(=O)C3CC3)C4)=O)ccc2c1 C(Cn1cc(-c2cccs2)nn1)(CC(C)C(C)C)N(C1C2CC3C(C2)C13)CC C1(C(=O)NCC(C(C)O)O)CCC(C)(C)N(C(=O)C(C(C)(C)C)N(C)C)C1 c1(OC)cc(C(=O)NCC(F)CNC(=O)C(C(C)O)N(C)C)cc(Cl)c1O N1(C(c2nccc(CC)c2)=O)CC(OC)CC1(C)CNCc1cc(C)cc(C)c1 C1(CC)CCC(O)(C(=O)NC2CC(CCNC(c3cnn(C(C)C)c3Cl)=O)C2)C1 N1(C(N2CCC(c3cn(Cc4[nH]nc(N(C)C)n4)nn3)C2)=O)CCS(=O)(=O)CC1 C(=O)(CC(C)(O)CCC)NC1CCN(c2ccc(C(C)=O)cn2)C(C)C1 CCC(C)CCC(O)CN1CCN(C(=O)OC(C)(C)C)C(C)C1 C1(NC(C(COC)C)=O)CC2CN(C(c3c[nH]cc(C)c3=O)=O)CC12 Cc1cc(C(=O)N(C2C3CN(C(c4nocc4Br)=O)CC23)C)cn1C(C)C Cc1cc(Br)cnc1C(=O)N(C)CCN(C(=O)CC1OCCC1(C)C)C N(C(=NCC(F)F)NCC(c1cccc([N+](=O)[O-])c1)SC)Cc1n(C)ncc1 CCCCC(C)C(=O)NC1(CCOC)CCN(C(=O)CC2CC(=O)NC2=O)CC1 C=C(C)C(C)(O)C(=O)NCC1CCN1C(C1(C(F)F)CCC1)=O C(=O)(C1Cc2ccc(F)cc21)NCCCOCCNC(C(c1cn(C)nc1)O)=O c1(OC)ccccc1C(=O)NCC(C(C)(C)C)NC(=O)CCc1cc(C)[nH]n1 c1(NC(CSCC)=O)ccccc1SC1(C)C=CCCC1 N1(C(CCN(S(C)(=O)=O)C)=O)CCN(C(=O)C=C(C)C2CC2)C2CCCCC12 C(=O)(CCN(C(=O)C(C)N(C)C)C)NCC1(C(NOCCC)=O)CC1 N1(C(CN(C)Cc2ccccc2)=O)CCC(N(C)C(C2CC3C=CC2C3)=O)CC1 N1(C(C2CC(NC(c3c(C)cn(C)c3)=O)C2(C)C)=O)CCS(=O)CC1C c1(C(N(CC(C)NC(=O)Cc2ccnn2C)C)=O)ccc(OCC2CCC2)cc1 c1(Oc2cn(Cc3cn(C4(OC)CC4)nn3)nc2)ccc2cnc(C)cc2c1 C12(NC(CN(C)C(N)=O)=O)CCCC1N(C(c1cc(C#N)c(O)nc1N)=O)CC2 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCCC(CCNC(C(CC)OCC)=O)CC1 c1(-c2cn(C3C(C)CN(C(c4ccc(F)c(F)c4)C4CC4)C3)nn2)cc(N)cc(F)c1 C(=O)(C(O)CC(F)(F)F)NC1CC(CNC(c2nsc3ccccc23)=O)C1 N1(C(C(C)(C)c2ccno2)=O)CCCC(CNC(=O)CSc2ccccc2O)C1 c1(CC)ccc(C(=O)NCCCCCNC(=O)Cc2cnccn2)c(F)c1 c1(C(=O)NCC2C(CNC(c3cc(C)c(C)nc3)=O)C2)cc(N)c(C)cc1Cl N1(C(=O)OC(C)(C)C)CCOC2(CCCN(C(=O)NCc3cc(F)n[nH]3)C2)C1 N1(C(C2(C)CC2Br)=O)CCOC2(CCCN(C(=O)Cc3cnns3)C2)C1 CCC(C(=O)NC1CCN(c2nnc(O)s2)CC1O)C(C)C N1(C(C=CSC)=O)CCC(C2(O)CN(C(=O)CCOc3ccc(O)cc3)C2)CC1 Cc1ccc(O)c(CN2CC3(CC3)CC2C(N2C3COCC2C3)=O)c1 c1(C(=O)NC2(CNC(c3c(OC)c(Cl)ccc3)=O)CC2)cc2ncn(C)c2cn1 c1(C(N2CCC(C)C(NC(C3CS(=O)(=O)C3)=O)C2)=O)cnc(O)n(C)c1=O CCCC(O)CC(=O)NC1CC(C)CN(C(=O)CCC(=O)c2cnn(C)c2)C1 c1(CC(=O)N(C(C(=O)N(C(C(C)SC)C)C)(C)C2CC2)C)ncccc1F CS(=O)(=O)c1nc(N2CCC(NC(=O)COC3CC=CC3)C23CCC3)cc(Cl)n1 c1(C(C(=O)NC2CCN(C(c3cnsc3)=O)CC2)(F)F)cc(Cl)ccc1F c1(C(=O)NCC(c2ccccc2)C)sccc1CNC(=O)CCc1ncnn1C c1(NC(CC)C(C)C)ccc(NC(N2CCC(O)CC2)=O)cc1F CCC(C)CCC(=O)N(CC(=O)NC1CCC(N(C)C)CC1)CC1CC1 c1(CC(=O)N(C)CC2N(C(CN3C(C)CC3)=O)CCOC2)noc2ccccc12 C(=O)(C1CCC(C)(C)c2ccccc21)Nc1c2scc(C)c2ncn1 C1(C#CC(=O)N(CCN(C(C2CC3C=CC2C3)=O)CC)CC)(CC)CC1 C1(NCc2c(C(C)C)n(C(C)C)nc2)NC(=O)CC1(C)C c1(C(=O)NC(CCCC)CNC(c2ncc(N)cc2C)=O)cc(C)cc(C)c1C C(=O)(C(O)CC[S+](C)C)N1CCC(N(C(=O)COCC2CCC2)C)C1 Cc1cn2c(n1)C(C(=O)N1CC(NC(=O)C=CCO)C(N=[N+]=[N-])C1)CCC2 Cc1cc(N2CCC(N)CC2C)c(S(N)(=O)=O)cc1[N+](=O)[O-] c1(C(C)C(=O)NCCC2(NC(C34CC(C)C3C4)=O)CCCC2)ccccc1Cl c1(C(=O)NC2CN(C(=O)NCc3cccs3)CC2O)cnc2c(F)cccc2c1 C1(n2c(C(=O)O)ncc2)CCN(CCC2CCCCO2)CC1 C1(C(C)(C)O)(CNC(=O)CSc2cn[nH]c2)CN(C(C2(C)CCOC2)=O)C1 N1(C(=O)CNc2ncccn2)CCN(C2CCN(C(C3CCOC3)=O)CC2)CC1 S(=O)(=O)(c1cccc(N2CCCC(C(F)(F)F)C2)n1)NCCC(=O)NCC C1(C(C)Nc2n(CC)ncc2)COCCN1Cc1ccccc1 C1(C)(CNC(CN(C(C)C)C)=O)CCN(C(c2ccc(Br)cc2Cl)=O)CC1 c1(C(=O)NCC23N(C(C)=O)CCC2CCCC3)cc2ccccc2c(O)n1 C(N=c1[nH]c(=NCCCCS(N)(=O)=O)[nH]c2c1COC2)C1CCC(CC)O1 C(=O)(N=c1ccn(C2CC2)[nH]1)C1N(C(c2ccc(CC)cc2)=O)CC(C)CC1 C1(CNC(C(c2cscn2)N(C)C)=O)CN(C(=O)CC2CCCC(C)O2)CCO1 CCCC(CNC(c1ncoc1CNC(c1ccoc1)=O)=O)OCC Cc1cc(C(N2CCC(C)(NC(=O)Cn3ccnn3)C2)=O)ncc1Br C1(C(N(C2CCC(C(N3CCOC(C4CC4)C3)=O)C2)C)=O)CC2C=CC1C21CC1 C(CCC(=O)N(C)CC1(CSC)CN(C(=O)C=CC(=O)N(C)C)C1)OCC c1(C(C)=O)cc(CN2CCC(CC(=O)Nc3nnc(C)o3)CC2)ccc1F N1(C(c2c(CC)occ2)=O)CC2(C1)CN(C(c1cnn(C)c1Cl)=O)CCO2 c1(C(=O)NCC2C(NC(C3C(C)C3)=O)C2)cccc(-n2cccn2)n1 C(Cc1ccccc1)(C(=O)N(C1CCCNC1)CC)NC(CCC)=O CCCCCC(C)CC(=O)NC1CC(F)(CNC(c2cnc(C(C)(C)C)o2)=O)C1 N#Cc1cc(S(=O)(=O)N2CCCC(O)(C(=O)O)C2)ccc1C(=O)O N1(C(CC(CC2CC2)NC(c2ncc(OC)nc2)=O)=O)CC2(CNC(=O)N2C)C1 Cc1cc(C)c(C(=O)NC2CCN(C(c3cc(C4CCCC4)[nH]n3)=O)C2)c(S)n1 c1(OCC)cc(C(F)(F)C(=O)NC(C)CCCNC(C2CC2CF)=O)ccc1C C1(CNC(CCc2ccc(CC)s2)=O)CCCCN1C(=O)C(C)CC1CCCC1 C(C(C)(CC(C)C)NC(=O)Cc1ccc(CC(N)=O)cc1)NC(CC(=O)OC)=O Cc1c(C(=O)NC(C)(CNC(C2CC2F)=O)C(C)C)nnn1C C(=O)(CCC(=O)N1CCCC(NC(=O)CCCc2cnn[nH]2)C1)OCC c1(C(N2CC3C(C(=O)OC)C3C2)=O)n[nH]c2cccc(NC(=O)NC)c12 C(C)(CC(=O)NCC1C2CC1N(C(=O)C=Cc1cc[nH]c1)C2)(C(F)F)N(C)C C(N=c1[nH]c2ccccc2o1)C1(O)CCCN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 c1(C(=O)NCCC(C)NC(=O)Cc2nnc(O)s2)cc(Cl)cc(Cl)c1 C1(C(N(C(CC)C)C)=O)CCC(n2cc(C3CCCCO3)nn2)CC1.C(CNC)N N1(C(c2n(C)cc(C#N)c2)=O)CC2CCC1CN(C(=O)CCc1cc(Cl)no1)C2 N1(C(C2CC(=C)C2)=O)CC2COCCC2(NC(=O)Cc2cc(F)cc(Br)c2)C1 C1(NC(CCC(=O)NCCCOCCC(C)C)=O)CCC(C(F)(F)F)N(C)C1 N#CC(C(=O)N1CCCC1COCc1ccccc1)c1nccs1 N1(CC(C2CCOCC2)OC)C(=O)CN(CC(n2cc(Br)cn2)OC)C1=O C1(c2n(C(CC)(C)C)nnn2)(NCCn2cnnn2)CC2CCCCC12.SCC N1(C(CCN(C(C2CC(SC)C2)=O)C2CC2)=O)CCC2(CCOCC2)C1 N1(S(=O)(=O)c2ccon2)CCc2cc(F)ccc2C1 C(=O)(CCC(C)NC(c1cnn(C)c1N)=O)NCC(C)N(C)C1CC1 c1(C(=O)NCCC23CCC2CN(C(=O)C=CCO)C3)[nH]nc2ncc(Br)cc12 C(c1ccccc1)=CC(=O)N(C1CCN(n2cccn2)C1=O)CC#C C1(C(N2C(C(N3CCn4ccnc4C3)=O)C=CC2)=O)C2Sc3ccccc3C12 c1(C(N(CCNC(c2cnn(CCOC)c2)=O)CC)=O)cc(Cl)sc1Cl C(=O)(C1CC(=O)c2cccc(OC)c21)NCC(C)NC(CCC=C)=O c1(C(=O)NC2C3CN(C(C4CC(=O)NC4=O)=O)CC32)ccc2nc[nH]c2c1F c1(CCC(=O)NCCN(C)C(C2CC2Cl)=O)ccc2ncsc2c1 C(=O)(C1=CCCOC1)NCCNC(C12C(CN(C(C(c3ccccc3)C)=O)C1)C2)=O C1(C(N2CCN(C(CC(C)C3CC3)=O)C(CO)C2)=O)CN(S(=O)(=O)N(C)C)C1 Cc1c(C(=O)NCCNC(c2cnc(C3CC3)s2)=O)c(Cl)nn1C C(=O)(CCCC(=O)NC(C)C)N(CC(C)NC(CCC=CC(C)C)=O)C S(=O)(=O)(c1cc(Br)c(F)cc1F)N1C(C)(C(=O)Nc2c(Cl)ccc(OC)n2)CC1 c1(CC(=O)NC(CC=C)CNC(=O)C2CC2)cc(Br)ccc1C N1(CCCN(CC=C)CC2(c3ccccc3)CCC2)C(=O)CCN(C2CC2)C1=O c1(OCC(=O)NCC(C)(C)Cn2cc(C3(C)CCCO3)nn2)ccc(F)nc1 c1(CC(=O)NCC2CCCC(NC(=O)CSC(F)(F)F)C2)cccnc1Cl CC(C)CC(C(=O)N(C(C)C(=O)NCC1CNC(=O)CO1)C1CC1)C(N)=O CC(C)(C(=O)NCCCC1(NC(=O)CC2(C)CC2(F)Cl)CC1)c1cccs1 C1(C(=O)NCC(=C(C(=O)NC(CC)(C)C)C)C)CCCC(CF)C1 c1(C(N2C(CC(=O)NCC(C)(C)C#N)CC(F)C2)=O)c[nH]c2ncccc12 c1(NCC2CCC(c3c(F)cccc3)CC2)ncnc2ncnc(I)c12 CCN=c1[nH]cc(C(=O)NC(CNC(c2cnc(C3CC3)[nH]2)=O)C2CC2)s1 c1(CC)cccc(OC)c1C(=O)NC12CC(NC(c3cc(Cl)cnn3)=O)(C1)C2 c1(CC(=O)N(CC(C)NC(=O)CC2CC(O)C2(C)C)C)cccc(F)c1F C(=O)(C(O)CC(N)=O)N1CC(CCNC(C=C(C)C)=O)OCC1 c1(C(=O)OC(C)(C)C)ccnc(OCc2ccccc2)c1.S1(=O)(=O)CCCN1 c1(CCC(N2CC(N(C)C(C3C4CNC(=O)C34)=O)C2)=O)cc(Br)ccc1F C=CC1(C(=O)NC2CCC(C)(CNC(=O)C=COCC)C2)CCOCC1 c1(C(N(CC(C)C(F)(F)F)CC)=O)ccc(O)c(C)c1C C(=O)(CCP(C)(C)=O)N1CC(OC)C(C(=O)N(C)CC2CCN(C)C2)C1 c1(CC)ccc2c(c1)C(NC(C13CCCCC1OCC3)=O)C(=O)N2C C1(CNC(C2(NC(CCCOC(C)=O)=O)CCOCC2)=O)CC1C1CCCC1 c1(C(=O)NC2C=CC(CNC(c3cnnn3C3CC3)=O)C2)cc(Cl)cnn1 c1(C(=O)NCC2CCCN(C(c3cc(C(C)=O)cn3C)=O)C2)c[nH]cc(F)c1=O c1(C(N2CC3CC2CN3Cc2cnc(Cl)s2)=O)cc2ncccn2n1 CC(C(=O)NCc1ccc(CNC(c2cnc(S)[nH]2)=O)c(F)c1)C(C)(C)C c1(C(=O)NC2C3(CCN(C(C(C)=CC)=O)CC3)C2)nn(C)c2ccccc2c1=O Cc1cn2cc(C(N3CCC4(CCC4NC(=O)C4CC4)CC3)=O)cc(C)c2n1 c1(C(N2CCC(NC(CC(=C)C)=O)CC2C2CC2)=O)ccnc2c1ncn2C Cc1cc(C(N2CCC(O)(CCNC(c3ccco3)=O)CC2)=O)c(Cl)cc1F C(N=c1cc[nH]cc1S(=O)(=O)NCc1ccc(COC)cc1Cl)C1CC(CC)C1 c1(CNC(=O)NCC(=O)NCC#CCNC(C2(C)CCC2)=O)ccccc1 Cc1cc(NC(=O)CCC2CCCN2C(=O)Cc2ccccn2)cc(C)c1 N1(C(CC2CC(=C)C2)=O)CCC2CN(C(C3(C4CCCO4)CC3)=O)CC12 N1(C(C=CCCC)=O)CCC(NC(C2CCC(C(C)(C)C)O2)=O)C(C)(C)C1 c1(OC)nc(C(N2CCC(NC(c3ccc(C)c(C)c3)=O)CC2C)=O)cc(O)n1 CC1Cc2cccc(C(=O)NC3(CNC(=O)C4=C(Cl)CCOC4)CC3)c2O1 C(=O)(C(C)CC(C)C)N(CCCNC(C(=Cc1cnc[nH]1)C)=O)C1CC1 CCCCC(=O)C(=O)NCC(CC1CCCC1)C(N1C(C)CCCC1C)=O N1(C(CCC(=O)N(C)C)=O)CCCCC(NC(c2ccc(CN(C)C)cc2)=O)C1 N1(C(C(COCC)C)=O)CC(C)(C)CCC1CNC(c1cscc1C(F)(F)F)=O C(CS(=O)(=O)CC(=O)NCC1CN(C(c2nnc3n2CCOC3)=O)CC1C)OC N1(C(Cc2c(CC)cccc2)=O)CC2(CCN(C(c3cncc(N)c3)=O)CC2)C1 C=C1CCC(CNC(C2CC3(C2)CC3NC(=O)C(C)OCC)=O)CC1 CC1CC(C(=O)NCCN(C(=O)CCN2CCC(O)CC2)CC2CC2)CC(C)C1 c1(CC(=O)NCCCCCCNC(CSS(C)(=O)=O)=O)ccc2cccnc2c1 c1(N2CC3CN(C(C4(C(=O)OCC)CCO4)=O)CC3C2)ccc2nccnc2n1 CC1=C(F)CN(C(C2C=CCN2C(c2cc(C)nc(C)n2)=O)=O)CC1 c1(C(=O)NCCCN(C(C2(C(=O)NC)CC2)=O)C)cn(C)c(=O)nc1O CCCCC(O)C(C)C(=O)NCC(C)CN(C)C(c1cnc2ccnn2c1)=O N1(C(C(C2CN(C(C3(C#N)CCOC3)=O)C2)OC)=O)CCOC(C)(C)CC1 c1(C(N2CC(F)CC(NC(C3CCCCC3)=O)C2)=O)c[nH]c2ccc(Br)cc12 N1(C(c2ccc(C)nc2)=O)CC(O)CCC1C(N1CCCC(CO)C1)=O N1(C(C2CCC(CC)O2)=O)CC(CNC(c2cc(C3CC3)on2)=O)CC1(C)C N1(C(C(c2ccc(C)s2)C)=O)CC(NC(c2csnn2)=O)CC(C)(C)C1 c1(C(=O)NCC2(F)CC(NC(C3(C)CCCCO3)=O)C2)cc(N)ccc1Br c1(C(C)CN(C(=O)CNC=O)C)cccc(F)c1 C1(NC(c2nc(CC)oc2)=O)CC(NC(=O)CN2CC(=O)NC2=O)CC1O N1(C(c2cnc(C)[nH]2)=O)CC(CNC(c2n[nH]c(C)c2Br)=O)C2(CCC2)C1 C1(NC(c2ccsc2Cl)=O)CC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 N1(C(C2(CC#C)CCC2)=O)CCC2(CC1)CC2C(=O)NC1CCC(O)(CC)CC1 CCC(COC)C(=O)NCC1(C(N)=O)CN(C(=O)Cn2nnc(C)n2)C1 c1(CNC(C(c2ccsc2Br)N(C2CCC2)C)=O)cccc(Br)c1 c1(COC)nc(OC)cc(N2CCC(CCNC(=O)CNC=O)(OC)C2)n1 N1(C(=O)CSC(F)F)CC2CC(NC(C3(C4CCCO4)CC3(F)F)=O)CC2C1 CCCCC(O)C(=O)Nc1cccc(-c2c(OC)cccc2O)n1 N1(C(COCc2onc(C)n2)=O)C2CCCC1CN(C(=O)C(F)=C1CCC1)CC2 c1(C(=O)NCCC(=O)NC2CC2(F)C(=O)O)c(F)cccc1F C1(CNC(c2c(C)cno2)=O)CCC12CCN(C(c1nocc1Cl)=O)CC2 C1(C)(CNC(CCOCC(C)C)=O)CC(NC(C2CCC(O)C2)=O)C1 N1(C(CC=CCNC(CCCCCSC)=O)=O)CCCCC(C)(F)C1 C1(N(C(CCNC2C(CC)C2)=O)C)CCN(C(C2CN(C(C)=O)C2)=O)CC1 C1(NC(C2CC(=C)C2)=O)CC(CNC(c2c[nH]nc2OC)=O)C12CCC2 c1(CNc2ccc(-c3n(CCC)ccn3)nc2)cc(CO)cc([N+](=O)[O-])c1 c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)cncc2[nH]ccc12 CC(C)(CC(F)(F)F)C(=O)NC1CCC1NC(=O)CCc1cccnc1Cl C(=O)(CC(C)C(C)(C)C)N1CCC(O)(CNC(C=COCC)=O)C1 C1(C(=O)NC(c2nc(=O)o[nH]2)C)(NC(=O)CCN(C)C)CC1(C)C C(=O)(C1=NOC2COCC12)N(C1CN(C(=O)CCn2cccn2)CC1(C)C)C N1(C(C=CC=CC)=O)CCCCCC1CNC(=O)CC1CSC1 C1(C(=O)NCC2(OC)CCC2)CC(NC(=O)CC=C(Cl)Cl)C12CCC2 c1(C(N2C(CNC(c3cnn4cc[nH]c34)=O)CCC2)=O)cccn(O)c1=O c12ccc3c(c1)N(CCS3)C2=O.C1(CNC)CCN(C(=O)COC(F)(F)F)CC1 N1(c2c(C(=O)OC)cc(C)cc2)CC2CCC1C1CN(C(C)=O)CC21 c1(-c2cnc(CNC(c3ncc(C#C)nc3)=O)nc2)ccc2c[nH]nc2c1 C1(O)(CNC(CC(CC)C)=O)CCCN(C(c2cc(Br)cnc2N)=O)C1 CCC(CC(C)C)C(=O)NCCN(C(C1C(F)(F)C12CC2)=O)CC1CC1 N1(C(c2c(CCC)[nH]cc2)=O)CCCC(CNC(C2CCC(C)(C)C2)=O)C1 C1(C(N2CC3C(CCNC(C4CC=CC4)=O)(CC3)C2)=O)CCCCC(F)(F)C1 c1(C(C)=O)ccc(C(=O)NC(CC2CCCC2)C(=O)N(C)Cc2ncc[nH]2)[nH]1 C(=O)(CC1COc2cc(O)ccc21)N(C1CC(NC(CCC=C)=O)C1)C c1(N2CC3C(C(F)F)(C3)C2)nccc(Sc2ncc(-c3ccccc3)[nH]2)n1 c1(C(=O)NC(C(C2CC2)OC)C)cc(CCNC(C2CC2(F)Cl)=O)on1 c1(CCNC(c2cnc(C)o2)c2nnnn2C(C)(C)C)c(C)noc1C CC1=C(C(=O)N2CC(NC(c3cccc(CO)n3)=O)CC2(C)C)SCCO1 C1(C(=O)NCC2C=CC(NC(Cc3n[nH]c(=NC)s3)=O)C2)CCCC12CC2 c1(CCC)nc(C(=O)NC(C)C(=O)N(C)Cc2nncs2)co1 c1(CC)cccc(C(c2nnnn2C2CCOC2)NCCCCCOC(C)C)c1 CCCCC(CNC(=O)C(c1ccc(Cl)cc1)=O)NC(c1cnn(C)c1)=O CC(C)C(C(=O)Nc1cncc(C(=O)NCCC2CCOC2)c1)c1ccccc1 CCCC(CC)CC(=O)NCC(CNC(c1ccc(CO)c(Cl)c1)=O)CO c1(C(N2CCC(NC(=O)C=CSCc3ccco3)(CO)C2)=O)c(F)ccc(F)c1Cl N1(C(CCCC(C)=O)=O)CCC(O)(C2(NC(c3cc(Br)co3)=O)CC2)CC1 C1(CNC(C(C)OCOC)=O)CC2CCC(C1)N2C(=O)CCc1ccoc1 C1(OC)CC(CN)N(C(C2CC3(CC3)CO2)=O)C1.C1(=O)C(C2CC2)N1C CNS(=O)(=O)N1CCN(C(=O)C(Cc2ccco2)NC(=O)OC(C)(C)C)CC1 N1(C(C(COC)C)=O)CCCC(C2CC2NC(c2cccc(C)c2F)=O)C1 N1(C(C2C3(CC(NC(C(C)N(C)C)=O)C3)C2)=O)CCCC(C)(C)C1 C1(CC(=O)NCC#CCC)CN(C(c2cc(F)ccc2O)=O)CC12CC2 Cc1sc(S(N)(=O)=O)cc1C(N1CC2(CC(NC(=O)C=C3CCC3)CO2)C1)=O c1(CCC(=O)NC2C(NC(C(C)NC(CC)(C)C)=O)C2)ccc(OC)c(O)c1 C1(NC(c2cc(SCC)ncc2)=O)CCCCN(C(C2(CO)CCCO2)=O)C1 C(=O)(C1CCc2nccn21)N1CC(CCC)N(C(=O)CC2CCOCC2)CC1 NS(=O)(=O)c1cccc(CCC(N2CC3(CNC(=O)C3)C2)=O)c1 Cc1ccc(CNC(c2ccc(CO)o2)=O)cc1.C1(NC(=O)C2CC2)CC(OC)C1 C1(C(N(C)CC2(CNC(c3cnco3)=O)CC2)=O)CCCCS1(=O)=O C12(C(=O)NCC3(C(=O)NCCC(C=C)(C)C)CC(=C)C3)CC3CC(CC(C3)C1)C2 C1(CNC(c2c(SC)snn2)=O)CCC(N(C)C(c2nnsc2C)=O)CC1 C1(CNC(C2N(C(C)C)CCC2)=O)CCCCN(C(=O)C(C)c2cccs2)C1 C1(C(=O)NC(C)(C)CCNC(c2ccnn2C2CCCCC2)=O)CCC12CCC2 N1(C(COc2ccc(OC)cc2)=O)CC2CC1CC2NC(=O)CC(C)F C(=O)(CCCCCS(N)(=O)=O)NC(CC)CN(C)C(c1ncoc1C)=O c1(C(N2C(CNC(c3ccc(OCC)c(O)c3)=O)CC2)=O)cc2ccccc2o1 Cc1ccc(-c2cn(-c3ccccc3C(=O)N(C)C(C)C)nn2)c(C)n1 N1(C(c2ccc[n+]([O-])c2)=O)CC2(CCCN(C(c3ncncc3Br)=O)C2)C1 N1(C(c2cc(C)ns2)=O)CC=C(CC(=O)NCC2(O)CCC(C)C2)CC1 c1(N2C(C)CN(C(=O)CC3(c4ccccc4)COC3)CC2)ccn2nccc2n1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2(CC1)CC2C(=O)NC1CCCC(O)C1 c1(N2CC(C)S(=O)(=O)CC2)cccc(S(=O)(=O)NC2CSCC2C)n1 c1(C(N2CC(CNC(c3ncsc3Br)=O)C2)=O)c[nH]c2ncc(Br)cc12 C1(C(N2CC3CC3(CNC(C3(CO)CCC3)=O)C2)=O)Cc2nccn2C1 CC(C)(C)C(=O)C(=O)NCC1(CNC(C2(OC)CCCOC2)=O)CC1(F)F S(=O)(=O)(c1ccc2ccccc2c1)NS(=O)(=O)Cc1noc(Cc2ccc(F)cc2)n1 C1(NC(C2C(CC)C2)=O)C2CCCN(C(=O)CCOCC(C)(C)C)C2C1(C)C Cn1nc(-c2cccnc2)cc1C(=O)NC1CC1NC(c1ccon1)=O CC#CCC(C(=O)OC(C)(C)C)NC(=O)NCc1c(OCC)cccc1C C1(C(=O)NCc2nc(C(=O)OC)sc2)CCCCN1C(c1ccc(F)nc1)=O c1(C(N2CC(C(=O)NCC(CSC)(C)O)C(C(C)C)C2)=O)ccc(C)cc1O N1(C(C2(CC#C)CC2)=O)CCN(C(=O)Cn2cc(C3CCOC3)cn2)C(CC)C1 C1(C)(CNC(C(COC)OC)=O)CN(C(=O)CCN2C(=O)CCC2=O)C(C)(C)C1 Cc1ccc2c(c1)CN(C1CCN(C(=O)OC(C)(C)C)C(C)C1)CCO2 N=c1ccc(C(=O)NCC2CCC(NC(C3C4CC5C(C4)C35)=O)CC2)n[nH]1 c1(NC2CCN(C(CC(c3ccc(C)cc3)C)=O)C2)cc2nncn2cn1 c1(C(N(CCNC(=O)Cc2[nH]cnc2C)CC)=O)cc2c(Cl)cccn2n1 C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(C(C)(Cl)Cl)=O)O C12(C(N3CC4CCN(C(c5nn(C)c(O)c5)=O)CC43)=O)CCCC(=O)N1CCC2 c1(NC(COC)C)c(F)ccc(Cl)c1CO.c1(CO)nc(C(C)(C)C)no1 CC(C)(C(=O)NCc1cc(C(=O)NC2CCN(C(C)(C)C)C2)n[nH]1)C(F)F Cc1nc(NCc2nc(C3CC3)cs2)cc(=NCC2(C)C=CCCC2)[nH]1 N1(C(C(CC)NC(N)=O)=O)CC(=O)CC1C(=O)NCC12CCC(CC1)O2 c1(OC)ccc(CNC(=O)C(C2CC=CCC2)NC(=O)C(=O)NC(C)C)nc1 C1(NC(=O)CCF)CC2CC(C1)CN(C(=O)Cc1ccc(F)cc1Br)C2 C1(NC(=O)CCc2cnc[nH]2)CCCN(C(=O)C=CC2CCCCCC2)CC1 CC1=C(C(=O)N2CC(NC(C3(C(C)(F)F)CC3)=O)C(C)(C)C2)CCO1 c1(OCC(C)(C)N2C(CC3CCCC3)C(=O)NCC2)cccc(C)c1.CCC(C)C C1(NC(COC2C(C)CCCC2)=O)CCSC12CN(C(=O)C(C)(C)C1CCC1)C2 c1(OC)c(C)ccc(C(=O)NC2CCCCCC2NC(=O)CN(C)CCO)c1F C1(NC(CCN(C(C)=O)C)=O)CN(C(=O)CCNC(=O)N(C)C)CCC12CCC2 C1(c2nnnn2CC(F)F)(OCC=C)CCN(CC2CCC(C(N)=O)CC2)CC1 c1(CC(=O)NC2C(NC(c3c(CCC)nns3)=O)CC2)ccc(F)cc1F C#CCC(C)(CNC(C1(C)CN(C(=O)CC(C)C)CC1C)=O)CO C1(NC(C(COCC)C)=O)CC12CCN(C(c1snc(Cl)c1Cl)=O)CC2 c1(NC(C(=O)NCc2c(C)cccc2)=O)ccnc2c1CCO2 C(CC(C)(C)C)(C(=O)N(CCC(C)O)C)NC(CC1CCC(C)CC1)=O C(=O)(C(C)CCCC)NC(CCOCC)C(=O)NC(C)(C)CF C1(CNC(CCC2(C)CC2)=O)CC12CCN(C(C1CC3(CCO1)CC3)=O)CC2 C1(C(=O)NC2C(NC(CC(C)CF)=O)CCC2)CC2CC(C1)CC(F)(F)C2 Cc1n[nH]cc1CC(=O)NC(C)C(C)(C)NC(=O)C=CCOCc1ccccc1 C(=O)(C1=CCCC1)N1CCC(CNC(CN(CC(=O)NC(C)C)C)=O)C1 CC(c1ccccc1F)=CC(=O)NC(Cc1ccccc1)CCC(=O)O CCC(C)(CCNC(=O)C=Cc1ccnn1C)NC(CC1CCN(C(C)=O)C1)=O C(CC(C(=O)N1CCC1C)NC(=O)Cc1cccs1)=CC N1(C(C(=O)NC(C)C)=O)C(C)CC2CN(C(c3ccc4ncncc4c3)=O)CC12 C1(CC(N2CCOC(CC3CCN(C(=O)CC4CC4)CC3)C2)=O)CC2(CC2)CO1 C1(N(C)C)(CNC(c2ccnnc2O)=O)CCCCC1.C12C=CCN1C2=O c1(C(=O)NCCn2cc(CN(CC)CC)nn2)c(O)cccc1O N1(C(C=Cc2n(CC)ccn2)=O)CCCC(NC(=O)C=Cc2nccs2)C1C C1(CC(=O)NC2(c3ccccc3)CC2)CC2(C1)CN(C(C1CCS(=O)(=O)C1)=O)C2 C1(CC#C)(C(N2CCC(CN(C)C(C3CC(C)(F)C3)=O)C2)=O)CCOCC1 O=C(C#Cc1ccc(Cl)cc1)N(C1CC2CNC1C2)CCc1ccc(Br)s1 CCCC(C)(O)C(=O)N(C1CC(NC(=O)CCCc2ccc(C)cc2)C1)C Cc1cccn2ncc(C(=O)NC(CNC(=O)C(F)C(C)C)C3CCC3)c12 c1(N(C)CC2NC(=O)CC23CNC3)c[nH]c2c(F)c(Cl)ccc2c1=O Cc1ncnc(C(N2CCC(C(C)(C)NC(c3c[nH]cc(F)c3=O)=O)C2)=O)c1C c1(NC(C2CC(C)CN2Cc2ncccc2O)=O)ncc(I)nc1Cl c1(C(=O)NC2(CNC(=O)CC3(O)CCOC3)CCC2)sc(Cl)cc1Cl CCC(CC)CCC(=O)NCC1CCN(C(=O)CN(C)C(N)=O)CC1C c1(C(C)C)ccc(C(N2CCCC2COC(C)(C)C)=O)nc1Cl C(c1nccn1CC)=CCO.C1(CCC)CC1C(NC(C)(C)C)N Cc1c(N)ccc(C(=O)NC2CS(=O)(=O)CC2NC(c2cocn2)=O)c1F C=CCC(C(=O)NC1(CF)CCN(C(=O)Cc2cccs2)C1)c1ccccc1 C1(C(N2CC(F)CC2CO)=O)CCCN(Cc2c(Cl)cncc2Cl)CC1 CCCCCCCCC(=O)N1CC2CC2(CNC(=O)Cc2cc(C)cs2)C1 CC1CCC(NC(c2ccc[nH]2)=O)CN1C(c1cc(Cl)ncc1O)=O Cn1nc(Br)c2ncnc(NC3CC(CNC(C4CCC(=O)N4)=O)CO3)c12 N1(C(C=C(CCC)CCC)=O)CC(N(C)C(c2[nH]c(=N)ccc2C)=O)C2(CC2)C1 c1(OC)cccc2cc(C(=O)NC(C)CCN(C(=O)CNC(=O)C(C)C)C)[nH]c12 C1(c2cn(C)nn2)CCC(NC(=O)COC2CCCCCC2)CC1 c1(CC(C)C(N(C(c2ccc(F)nc2)C)C)=O)ccc(F)cc1F C1(NC(CCN(C)CC)=O)C(CNC(=O)Cc2ccccc2Cl)CCC12CCC2 c1(CC)cc(C(=O)Nc2cccc(NC(=O)CN3CCCCC3C)c2)oc1CC N1(C(C2N(C(C(C3CCCC3)OC)=O)CC=C2)=O)CCC2(CCOCC2)C1 N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCN(C(=O)C#CC2CC2)CC(C)(F)C1 c1(C(N2C(CNC(C)=O)CC(O)C2)=O)nc(Cl)ccc1Cl S(=O)(=O)(C1CN(C(C2CCC2)=O)C1)N1CCN(C(C2CCCC(C)C2)=O)CC1 c1(C(=O)NC)ccc(C=CC(=O)NCCCCNC(C2CC(O)(C#N)C2)=O)cc1 C1(C(=O)NC2(CNC(c3c(C)n[nH]c3)=O)CC2)CC2CCCC12 C12(C(=O)NC(C3(O)CCN(C(CC(C)CF)=O)C3)C)CC3CC(C1)CC(O)(C3)C2 Cc1cc(C)c(C(N2CCC(CNC(c3cnn(C)c3C3CC3)=O)C2)=O)cc1N C=CC(F)(F)C(=O)N(CC(C)N(C(=O)OC(C)(C)C)C)C.C1(OCC(=O)N)CCCC1 C1(F)(CNC(C2(Cl)C(C)(C)C2)=O)CCN(C(c2cnccn2)=O)C1 C1(O)(CNC(c2cn(C3COCC3F)nn2)=O)CCN(C(=O)Cc2cnsc2)C1 c1(CN2C(CC(=O)Nc3cc(C#N)c(F)cc3)CCC2)ccc2[nH]nc(Br)c2c1 c1(N(C(C(C(C)C)n2cncn2)=O)CC(C)C)ccc(Cl)c(Cl)c1 C1(CC)(NC(=O)CN(c2ccccc2)C)CCCN(C(=O)Cc2ccc(C)o2)C1 CON=C(C(=O)NC(C)CN(C(=O)CCCC1CC1)C)c1ccco1 CCC(C)(O)C(=O)N1CCC1CNC(=O)Cn1nccc1C N1(C(C(CC)(C)CNC(c2cc(C)c(C)s2)=O)=O)CCCC2C(=O)NCC12 c1(C(=O)NCC2(CNC(C34COCC3C4)=O)CC2)nsc2ccccc12 C(=O)(C#CC1CCOC1)N1C(C(=O)Nc2cc(C)cnc2O)(COC)C=CC1 CCC(C)C(C(=O)NCCOC1(C)CCC1)N(C(=O)C1=CCCCC1)C c1(N(C(=O)C(O)C2CN(C(=O)CC=CC(C)(C)C)C2)CC)cccnc1 N1(C(C(CC)(C)C)=O)CCC2(NC(=O)Cc3cncnc3)CCCC12 C1(NC(C(CC=CC)C)=O)CCC2CN(C(=O)CNc3ccccc3Cl)CC2C1 N1(C(C=CCC)=O)CCC2(CC1)CN(C(c1ccnn1CCC)=O)C2 C(=O)(CCC(C)(C)F)N(C1CCCC(NC(c2nnc(C)s2)=O)C1)C c1(C(N2CCN(C(C(C)OC)=O)CC2c2nccn2C)=O)cc2c(s1)CCOC2 C1(NC(C(COC)N(C)C)=O)C(C)CN(C(c2cc3ccccc3s2)=O)CC1C N1(C(C2CC(CCC)C2)=O)CCC(NC(=O)C(C)CCC)C2(CCC2)C1 C1(CNC(C(c2cccc(C)c2)NC(=O)OC(C)(C)C)=O)CCOCC1(C)C N1(C(C(=O)Cc2ccc(F)cc2)=O)CC2(CC2)CC1CNC(=O)Cn1nccn1 C1(NC(C(C)SC)=O)COC2(CNC(=O)C(c3ccc(C)cc3)(C)C)CC1C2 c1(C(=O)NC(C2CCOC2)CNC(c2cccs2)C)cn(-c2cnn(C)c2)cn1 c1(C(N2C3C(C(=O)NCCC4C(C)CCCC4)C(C3)C2)=O)cc(F)c(F)cc1Cl N1(C(C(CCC)C#N)=O)CC2CCC(NC(=O)C(C)(C)OC(C)C)C2C1 c1(C(=O)NC2C=CCC(C(N3CCC(NC(C)=O)C3)=O)C2)cccc(O)c1C N1(C(C(=O)NC)=O)CCC(C)C1CNC(=O)CC1CCC(C)C1 C1(NC(=O)Cc2cc(C3CC3)on2)CN(C(=O)C2=C(Cl)CCC2)CCC1O C1(C(N2CCC(C(O)CNC(=O)C(C)CC#N)CC2)=O)(COC)CCOCC1 S(=O)(=O)(c1ccc(-n2nc(CO)nc2-c2coc(-c3ccccc3)c2)cc1)NC C=CCCC(C(=O)NCCNC)N(C(C)CS(C)=O)C CCN=C(NCC(C)SC)NCC1CCC(C(=O)OCC)C1 Cc1cccc(OCCC(N2CC3CC3(NC(c3cc(CO)oc3C)=O)C2)=O)c1 c1(C(=O)NC(C2(O)CCN(C(c3cc(Br)n[nH]3)=O)C2)C)noc2ccc(Cl)cc12 O=C1CCC2C(C(F)(F)F)C12.c12ocnc1C(=O)N1CC2C1.C1CO1 c1(C(C(=O)N(CCC)CCNC(=O)CC2CCC2)(F)F)ccc(C(C)(C)C)cc1 C(=O)(C1CCCc2n[nH]cc21)NCCC(C)NC(c1sc(CC)c(C)c1)=O c1(C(=O)NC(C2CCN(C(=O)CCC(CF)CF)CC2)C)cnc(O)n(C)c1=O C(=O)(C1=C(C)OCCS1)N(CCC(=O)N(C(CC)CC)C)C(C)C N1(C(CCc2c(C)noc2Cl)=O)CCC(NC(=O)C(O)c2ccsc2)C(CO)C1 CC1CCC(NC(c2cn3c(n2)SCC3)=O)CN1C(c1cc(C(F)F)nn1C)=O C(=O)(CCCCCOC)N1CCC(CCC(=O)NCC2CC(CC)C2)CC1 C1(NC(CC2(C)CCOC2)=O)CCCC(CNC(=O)CC2CSCCO2)C1 c1(CNC(c2c(Cl)ccc(CC)c2)=O)ccc2c(c1)CN(C(=O)C(C)CC)C2 c1(C2N(C(C3NCC(=O)NC3)=O)CCC2)nc2c(s1)CCC2 n1(CC)ncc(C(N2CCOCC2CNC(=O)C(C)c2ccon2)=O)c1C C1(C(=O)NC2C(NC(C(C)(C)Cc3cccc(Cl)c3)=O)CC2)NC(=O)OC1(C)C C#Cc1ccc(OCC(=O)NCCCCNC(C2CC(O)C2)=O)c(OC)c1 O=C(CC1=CCCC1)NCC1C2CN(C(=O)CCNC(=O)CO)CC12 c1(-c2n(CC)ccc2)nc(-c2cccc(OC)n2)nn1C1CCOC1C C1(NC(CSCC=C)=O)CC(CNC(=O)C(c2cccc(Cl)c2)(C)C)C12CCC2 c1(C(N2CCOCC(NC(C3C(C)CC(C)O3)=O)C2)=O)cccc2c1ncn2C Cc1ccn2nc(C(=O)NCCCC3(NC(c4cnnc(O)c4)=O)CC3)nc2n1 c1(CC(N2C(C)CC(NC(c3scc(C)c3)=O)C2)=O)cc2ccccc2c(O)n1 C12(C(=O)NCC3CCN(C(c4ccoc4)=O)C3)CC3CC1C2C3 CCC(C)(C)C(C(=O)NC(C)(CNC(c1cc[n+]([O-])cc1)=O)Cn1cccn1)OC CCCCC(CNC(c1ccc(-c2cccs2)s1)=O)NC(c1nc(O)sc1C)=O C1(F)(CNC(c2cnc(O)s2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1 c1(CNC(=NC)NCc2c(F)cc(F)c(F)c2F)cccc(S(N)(=O)=O)c1 c1(C(C)=O)ccc(NC(=O)Cc2cnc(NCc3ccc(Br)cc3C)s2)cc1Cl Cc1cnc(C)c(C(=O)NC2(c3ccccc3)CN(C(=O)CC3CCC3C)C2)c1 C1(CNC(C(C)(C)C)=O)CC2(CCC2)CN1C(C1CC=CCC1C(F)(F)F)=O N1(C(c2n(CC(C)C)ncc2)=O)CC2CCC(NC(=O)Cc3cn[nH]c3)CC2C1 C=CC(CC)CC(=O)NCCCCC1CCCN(C(=O)Cc2cn[nH]c2)C1 c1(C(=O)NC2C(NC(c3cc(C(C)=O)on3)=O)CCC2)c(C)[nH]c(C)c1C c1(OC)c[nH]c(C(=O)N(CCNC(C2CCOC(C)C2)=O)C(C)C)cc1=O c1(NC)ccc(C(=O)NC(C)CCNC(=O)CC2C(=O)ON=C2C)cn1 N1(CC(N2CC(C3CN(C(C(C)SCCCC)=O)C3)C2)=O)CCN(C)CC1 C12(C(=O)O)CCN(C1)Cc1cccnc12.c1(NCCC)ccc(NC)cc1.C(F)(F)F C(c1ccc(I)o1)=C(C(=O)NC(C(=O)NCCC)C)C C(=O)(CC(C)(C)F)NC1CC(CNC(Cc2nc(C)oc2)=O)C1 C1(C(=O)NC(CC#C)C)CN(C(=O)C2CC2)CCC1O c1(NC(=O)CC2CC3(CC3)C2)ccnc(Cl)c1C(=O)NC1CC(N(CC)CC)C1 Cc1cc(CN2CC(N3CCNC3=O)C2)cs1.C12(CC1)C(=O)NC2 N1(C(=O)CC(F)(F)F)CCC2CCN(C(C3(F)CC4(CCC4)C3)=O)CC2C1 N1(C(C=COCC)=O)CCC2(CCC(CNC(C3CN(C)C3)=O)O2)CC1 C(=O)(C1=CCSC1)NCc1nc(CNC(C(N2CCCCC2=O)(C)C)=O)sc1 C1(NC(C2CCN(C(C3N(CCC)CCC3)=O)C23CC3)=O)CCCCCCC1O c1(CNC(c2n(C(CC)C)nnn2)CC(C)C)cccc(Cl)c1Br c1(OC)c(C(=O)NC2C=CCN(C(C3CCC3C)=O)C2)cnc2c1cnn2C C1(C(C)C(=O)NCC(C)(C)F)CCCN(C(C2(CF)CC(=O)C2)=O)C1 N1(C(C(C(C)C)(C)O)=O)Cc2ccccc2CC1CNC(=O)CC1CCN(C)C1 Cc1oc(C)c(C(N2CC(NC(=O)CCc3cnoc3)C(C)C2)=O)c1C c1(C(N2C(CN(C(CCOCCOCC)=O)C)COCC2)=O)cccc(C)c1F C1(NC(c2cc(C)oc2C)=O)CC(O)CN(C(c2ccc(-c3ccco3)s2)=O)C1 C1(C#N)(CC(N2CCC(CC)(NC(=O)CCCN(C)C)CC2)=O)CCCCCC1 C1(C(N2CCC(NC(Cn3nnc(=N)[nH]3)=O)(CO)C2)=O)CCc2nc[nH]c2C1 C1(NC(C(CSC)(C)NC(C2CCCN(CC3CC3)C2)=O)=O)CC(F)(F)C1(C)C CS(=O)(=O)C(C(=O)NC1CCN(C(=O)C=CCN2CCCCC2)CC1)C1CC1 N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)CC2COCCN2C(C)=O)CC1C c1(C(N=c2ccn(C)[nH]2)=O)csc2c1CCN(C(c1cc(F)nc(F)c1)=O)C2 C(=O)(CC(C(C)C)Oc1ccccc1)N1CCC(NC(c2c(C)n[nH]c2)=O)CC1 C1(CNC(COCCOCC)=O)CNCCN1C(C1CN(C2CCOC2)C1)=O c1(CC)cc(CC(N2CC(CC(F)C(=O)NCCCCc3cnc[nH]3)C2)=O)on1 CCCCC(CC)CC(=O)N1CCC(N(c2nc(C)nc(=N)[nH]2)C)C1 c1(C(=O)NC(C)CNC(C2CCOC(=O)N2)=O)ccc2c(c1)NC(C)CC(=O)N2 C(c1ccc(F)cc1)=CC(=O)NC1CCC(NC(c2cccn2C2CC2)=O)CC1 N1(c2ncnc(=N)[nH]2)CCCC1C1CCCCN1C(=O)CC(=O)Nc1nccs1 c1(C(=O)OC)cccc(C(N)CNC(=O)COCC(N2CCCC2)C)c1 C1(C)(CC)CCN(C(=O)C(C)(C)CN(C)C(C2CCCOCC2)=O)C1 c1(C(=O)NC(C(=O)NCC(=O)OCC=C)C2CCOC2)ccnc(SCC)c1 c1(C(NOCC(C)(C)C)=O)cccc(Cn2cc(CN3CCCCC3)nn2)c1 C1(C(N2CC(CC(C)NC(COCCC=C)=O)C2)=O)CCOCC12CCCC2 C1(C(=O)NCC(CO)NC(C)=O)CCN(C(c2cc(CO)on2)=O)CC1 C1(NC(C2CCC(C)O2)=O)CCC(CNC(=O)Cc2ccsn2)CC1 CCCCC(C)C(=O)NC12CC1CN(C(c1conc1C1CCC1)=O)C2 c1(C(N2C(C(=O)Nc3cc(C)cc(O)c3)CC2C)=O)cc(C#N)ccc1C c1(C(N(CC(=O)N(CC(C)C)CC#C)CCOC)=O)ccccn1 N1(C(C2(n3ccnc3)CC2)=O)CCC(n2nccn2)CC1 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(c2cnn(C(F)F)c2)=O)C(F)C1 N1(C(=O)OC(C)(C)C)CCN(C(=O)Cc2ccccc2OC)CC1CC1CC1 C1(CNC(=O)CC2CSCCO2)C2CN(C(c3cccc[n+]3[O-])=O)CC12 N1(C(C2C(=C)C2C(=O)OC)=O)CCC(C)(NC(=O)C=Cc2ccc(C)s2)C1 C(=O)(C(=O)N=S(C)(C)=O)NC(CCCNC(CN1C(C)CCC1C)=O)(C)C N1(C(CCc2ccc(C(=O)OC(C)(C)C)nc2)=O)CC2CC1CC2(F)F C(=O)(CCCC(=O)N(C)C)NC1CC(C)N(C(=O)COCc2ccnc(O)c2)C1 CS(=O)(=O)c1ccnc(N(c2cc(O)ccn2)CC2CNC2)n1 N1(c2ccnc(C)n2)C2CCC1CC(CNC(=O)CC1(O)CCCN(C)C1)C2 Cc1cnc2ccc(C(=O)NC3(CNC(C4(Cl)CC4(C)C)=O)CC3)cn12 Cc1nn(C)cc1CN1CCC(C(N2CCC(NC(c3ccoc3)=O)C2)=O)CC1 c1(CC)cccc(C(=O)NCC2C=CC(NC(c3ccc(C4CC4C)o3)=O)C2)c1 N1(C(c2c(C)ncs2)=O)CCCCC1CCNC(=O)C(C(C)C)n1cccc1 Cc1nc(C(C)C)nc(N2CCC(n3ccc(NC(=O)CN(C)C)n3)C2)c1Br C12(C(=O)NCC3(NC(C4C5CCC(=O)C54)=O)CCC3)CCCC1C2(F)F N1(C(c2cn(CC(C)C)nc2)=O)CCCN(C(c2cnc(Cl)s2)=O)C(C)C1 c1(C(=O)NCC2(C(N)=O)CN(C(CSCCCC)=O)C2)ccc(OC)cn1 Cc1cncc(C)c1C(=O)NCC(C)(C(C)C)NC(C1CC2CCC1CC2)=O C1(F)(C(N2C(CCCC)CCC2)=O)CCN(Cc2c[nH]ccc2=N)C1 C(=O)(CC(O)CC(C)(C)C)NC1(C)CC(NC(CCCC)=O)C1 c1(C(C(=O)NCC)C)ccc(SCCN(c2ccc(OC(C)C)cc2)CC)cc1 c1(OCCCC(=O)NC(CC(=O)NCc2nc(C)sc2)C(C)C)ccccc1O CCCC(CCC)NC(=O)CCOCCN(C(=O)CC1CCC(=O)N1)C.CCO C=C1CCC(C(=O)NCCC2CCN(C(C3CC(OC(C)(C)C)C3)=O)C2)CC1 C1(NC(CSC(C)C)=O)COC2(CCN(C(C3(C#N)CC3(C)C)=O)CC2)C1 CCC(C)CCCCC(=O)NC1C(C)(C)C(NC(c2ocnc2C)=O)C1(C)C c1(CNC(C2CN(C)C(=O)O2)c2nnnn2C2CCC2)cc2ccnc(Cl)c2o1 N1(C(C(C)C2CC2)=O)CC2(NC(C3CC(=O)N(C(C)(C)C)C3)=O)CC2C1 Cc1ccc2sc(C(=O)NC(C)CNC(c3ccc([N+](=O)[O-])cc3Cl)=O)cc2c1 CCCC(C)CC(=O)NCC1(CCCNC(c2c(C)coc2C)=O)CCCC1 C1(N(C)C)CCCCC1(CO)NC(=O)CCCC(N)=O O=C(CCCCCc1ccccc1)NCCC1(CNC(C2SCCS2)=O)CC1 Cc1csc2ncnc(N3CCC(C)C3CNC(C3CCCCS3)=O)c12 N1(C(C(C)OCC)=O)CCCC(N(C(=O)C(c2ccccc2Cl)C)C)C1 CC(C)CC(C(=O)NC1CCOC(CNC(C2(F)CCC2)=O)C1)C(N)=O C12(NC(CCC3CCN(C(C4CCCC(C)C4)=O)CC3)=O)CCCN(CCC1)C2 CC(CCN1CCCCC1)C(=O)N1CCC1C1CCCCC1 C12(CCNC(C3N(CCC)CCC3)=O)CCC1CN(C(=O)Cc1c[nH]nc1O)C2 c1(OC)cncc(NC(C2CCCC2CNC(c2cnsc2)=O)=O)c1 C1(NC(C(Cn2ccnn2)NC(Cn2nnc(C)n2)=O)=O)CCN(C)CC1 c1(C(=O)N(CC2N(C(C(COC)OC)=O)CCCC2)CC)cc2ccsc2s1 c1(SCC)cc(N2CCN(C(=O)C(C)C(C)CC)CC2)nc(SC)n1 c1(COC)noc(COCC(C)CNC(c2cnn(CCN(C)C)c2)=O)n1 c1(SS)ncnc2[nH]cnc12.C1(C(=O)NCC(F)CO)CCCN(C(=O)CCN)C1 Cn1cccc(C(=O)NCC2(C(N3CCOC(C(N)=O)C3)=O)CC2)c1=O C(CN=c1nc(N2CCC3(CCC3)C(CO)C2)c2[nH]ccc2[nH]1)N(C)CC C(=O)(CCCCCC(C)O)NC1C(CNC(c2ccc(CC)cn2)=O)COC1 N1(C(C)C)CCC(C(=O)NC(C)(CNC(C2CC2F)=O)CO)CC1 CC(C)C(C)C(=O)N1CCC(CNC(C2CCCC(CF)C2)=O)CC1 CCC(C)(CC(=O)NCCSc1cccc(CNC(CC(C)O)=O)c1)C(=O)OC N1(C(C2C(C)(C)C2)=O)CCCC12CCN(C(c1cc3c(s1)CC(C)(C)C3)=O)C2 C(c1ccc(S(C)(=O)=O)o1)=CC(N1CC(C#C)C(NC(=O)NC)C1)=O C(C(C(C)(C)C)Nc1cc(C(F)(F)F)ncn1)NC(C1(CN(C)C)CCC1)=O c1(C(=O)O)cccc(-n2nc(CC3CCC3)nc2CC2CC2)c1 N1(C(C=C(C)C)=O)CC(C)CN(C(c2ccnc(O)c2Br)=O)C(C)C1 CC(CNC(=O)C(C)(C)n1cnnn1)(Cn1cccn1)N=c1cc(Cl)c(O)n[nH]1 O=C1CC2(CCN(c3nc(N4CCCSC4)nc4scnc34)C2)Oc2ccccc21 c1(NC(OC)OC)cc(Br)ccc1S(=O)(=O)NCCCCNc1cccc(Cl)c1 Cc1noc(C(F)(F)Cl)c1C(=O)N(C1CN(C(=O)C#CC2CC2)CC1F)C c1(C(N2CCC(N(C(C3CC3CF)=O)CC)C2)=O)ccc2cn(CC)nc2c1 CCC(O)C(F)(F)C(=O)NCCC1(O)CCN(C(c2cc(N)c(Cl)c(O)c2)=O)C1 CCC(CCC(=O)NCCc1ccncc1F)NC(C1CNC(=O)O1)=O CC#CCCC(=O)NC1CC(CNC(=O)CCCCC2CCCCC2)C1 C(=O)(C(C)(C)C(=O)NC)NC1CCC(C(N2CCC2(C)COC)=O)C1 CCC(C)(CNC(C1CCC(C)N1C(C12CCC(C1)C2)=O)=O)CO C1(C(N(C2CCN(c3ccnc(C(F)(F)F)n3)C2)CCC)=O)CCc2cncn2C1 N1(C(C(CC(C)C)F)=O)CCC2OCCN(C(=O)CCC(=O)c3cccs3)C2C1 c1(Nc2ccc(NC(C3CNC(=O)O3)=O)cn2)ccc2nccnc2c1 C1(C(N(C2CCN(C(=O)COc3ccc(CO)cc3)C2)C)=O)Cc2ccccc2C1 c1(CC)[nH]nc(C(=O)NC(CO)C(C)NC(=O)NC)c1Cl C1(NC(C2CCN(C)CC2)=O)CC(F)(F)CC1NC(c1ccccn1)=O c1(NC(C)=O)ncc(S(=O)(=O)NC2CN(C(c3nccnc3Cl)=O)CC2F)s1 N1(Cc2cccc(OC)n2)Cc2[nH]nc(NC(c3ncccc3Br)=O)c2C1 c1(C(=O)NC(CN(C(CC2N(CC)CCC2)=O)C)(C)C)cc(OC)cc(C)n1 C=CCC(CC)C(=O)N1CCN(C(c2cncc(C)c2Cl)=O)C(CCO)C1 c1(N2CC(NC(C3CCN(CCCCF)CC3)=O)C2)ccccc1[N+](=O)[O-] CC1CCCN(C(=O)CCN2CCN(C)CC2)C1CNC(=O)COC(F)(F)F C1(c2nnnn2CC(F)F)(NCC2(C)COC2)CC2CC1CC2F CCC(C)C(O)C(C)C(=O)N1CCC(N(C(=O)CCc2csnn2)CC2CC2)C1 Cc1cc(C(=O)NCCC2(O)CN(C(c3cn(C)nc3Cl)=O)C2)cc(C)c1F C1(C(=O)NCC(C)(C)CNC(=O)C(F)F)CC12C1CC3CCC(C1)CC2C3 c1(C(CNC(c2ccnn2CC(C)C)=O)NC(C(=O)NCC)=O)cccc(C)c1 C1(OC)CN(C(=O)C(O)COCc2ccccc2)CC1NC(C1CCCCCS1)=O C1(NC(CN(C)CC)=O)CCCN(C(c2ccccc2OC2CCC2)=O)C1 c1(NCC(CNC(CS(CCOC)(=O)=O)=O)O)ccc([N+](=O)[O-])cc1Cl C1(NC(CC#CC(=O)NOC2CCCCC2)=O)CC2CC3C(C2)C13 N1(C(c2cc(OCC)ncc2)=O)CC(NC(C2CC2C(N)=O)=O)C(C)(C)C1 c1(OC)nc(Cl)ccc1C(=O)NCCCC1(NC(C2CCCC2O)=O)CC1 CC1CCN(C(c2ccc[nH]2)=O)CCN1c1ccnc(C2CC2)n1 Cc1ncn(C)c(=O)c1C(N1CC(NC(C2(C#N)CC3(CCC3)C2)=O)C1)=O C1(OC)CC2(C1)CC(C(=O)NCC(C(C)(C)C)NC(C1CCC(F)(F)CC1)=O)C2 C=C(C)C(C)(C)C(=O)N1CC2CCC2(CCNC(=O)Cc2coc(C)n2)C1 N1(C(CC(CC)(C)C)=O)CCCN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1C N1(C(C(CCNC(CCn2ccc(C)n2)=O)O)=O)CCc2ncncc2C1 C(c1c(Cl)cccc1Cl)=CC(=O)N(CC(C)(C)NC(c1c(C)snc1)=O)C c1(OC)c(CC(=O)NC2CC(C)(C)C2)cc(Cl)cc1-c1ccccc1 C(=O)(CCCN(C)C)NCCCOCCNC(C1C(C(N)=O)C1)=O CCCCC(O)C(=O)NC1CN(C(=O)CCOc2ccccc2)CC1O CC1CC(CNC(=O)CC2CCCC2C)CN1C(=O)Cc1cccc(O)c1 N1(C(CC(CCC)C)=O)CC(NC(=O)Cn2ncc(Br)n2)CC(C)(C)C1 c1(C=O)cc(N)c(F)cc1C.Cc1ccc(C)cc1.N12CC=CC(C1)NC(=O)C2 C1(C(N(CC(C)NC(C=CCC)=O)C)=O)CC(=O)NC(=O)C1 C(=O)(CC1OCCc2ccsc21)N(C1CCN(C(C(CCC)CCC)=O)CC1)C N1(C(=O)OC(C)(C)C)CC2(CC(NCCc3cccc(Cl)c3Cl)c3nccn32)C1 C1(C(=O)NCc2cccc(NC(CC3CC(=O)OC3)=O)c2)CC2C=CC1CCC2 c1(C(N2CC(C(C)(C)O)(CNC(CCCCCC)=O)C2)=O)cc2n(n1)CCCO2 c1(COC)cc(C(=O)N(CC(C)SC)C)n[nH]1.C12(CC(C(F)F)C1)C(=O)N2 c1(N2CCCC(CCO)C2)nc(=NCc2csc(O)n2)[nH]c2ccsc12 Nc1cc(Cl)ccc1C(N1CC2CC(NC(=O)C(C3(O)CCCC3)F)C2C1)=O C(CC(=O)N(CC(O)CN(C(=O)CCc1cnn(C)n1)C)C)(C(C)C)OCC N1(CC(=O)NCC2CCCN(C(c3cncnc3)=O)C2)C(=O)C=CC1=O CCC(C)CN=c1cc[nH]cc1S(=O)(=O)NCCN1CC=CC1 c1(C(N2CC(CCNC(C(C(C)C)O)=O)C2)=O)cc2ccnc(Cl)c2s1 C1(CCNC(C(c2ccc(C)cc2)=O)=O)CN(C(C2(O)COC2)=O)CC(C)O1 c1(OC)cc(C(N2CC(CNC(=O)CN(C)C)C3CC23)=O)cnc1O CCCC(C(=O)NCCCC(CO)NC(=O)C(C)N1CC(C)C1)C(C)C C(=O)(CC1=CSC2=NCCN12)NC1C(C2CCN(C(c3cc(C)cnc3)=O)CC2)C1 S(=O)(=O)(c1c(C)cccc1Cl)N1C2CN(C(CCCC=C)=O)CC21 N1(C(CC2CCN(C(c3ccc(NC(C)=O)o3)=O)C2)=O)CCn2ncc(C)c2C1 Cc1ccc(N2CCCC(NC(C3CC(C)(F)C3)=O)C2)c([N+](=O)[O-])c1 C1(CNc2c(N(CC)CC)cccc2)C(=O)NCC(=O)N1C.C(C)(C)(C)N(C(=O)N)C c1(C(=O)NCC2CN(C(C=CCOC)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C1(C(=O)NCC2CCCCN2C(=O)CCc2ccnc(O)c2)OC2CCC1CC2 c1(OC)ccc(NC(=O)C(=O)NC(C)C(=O)NO)cc1S(C)(=O)=O CC(C)(C)C(C(=O)NCC1(O)CCN(C(c2cccs2)=O)C1)N1CCNC1=O c1(CC(N2CCCC(NC(C)C(=O)NC(N)=O)C2)=O)cc2ccccc2s1 CC1CC2(CCN(C(=O)CN3CCC(C)C3)CC2)CN1C(=O)CC1=CCCC1 C1(C(N(CCOC)CCNC(=O)CSCC(C)C)=O)CCCOC1C c1(CNC(=O)CC2CC2)cccc(-c2cnn(C3COC3)c2)n1 C1(O)(CNC(C(C)C(F)(F)F)=O)CC2CCC(C1)N2C(=O)CC1(C)CCC1 N1(C(c2ccc(CSc3scc(C)n3)cc2)=O)CCN(C)C(=O)C1C C12(C(NC[Si](C)(C)C)=O)CCCC1CCN2NC(C1CCC2(CCC2)C1)=O C1(NC(C(C)Cc2ccc(F)cc2)=O)CN(C(=O)C(O)C2CCC2)CC2(CC2)C1 c1(C2(C(=O)NC3CCC(NC(C4(OC)CC4)=O)C3)CCC2)ccc2c(c1)OCO2 C12CC3CCC1N(C3)C2=O.c1(NC(C(=O)NCCC(N)=O)=O)ccc(O)cn1 N1(C(CC(CC)C)=O)CCC2(CCCN2c2nc(C3CC3)ccc2C#N)CC1 CC1CCN(C(C2(F)CCOC2)=O)CCN1C(=O)CCc1ccc[nH]1 N1(C(c2ccns2)=O)CCC(C2CCN(C(c3cnc(C(F)F)s3)=O)C2)CC1 N1(C(C(COC)(C)O)=O)CCC(F)(F)C(CNC(C2(F)CCOC2)=O)C1 c1(C(=O)NC(C(C)C)CCN(C(=O)CCCF)C)ccc2c(c1)CN(C)CC2 Cc1sc2ncnc(N3CCCC(C)(CNC(=O)C=Cc4cnc[nH]4)C3)c2c1C N1(CC(=O)N(c2cccc(C)c2)CC)CCOC(C(=O)O)C1(C)C c1(C(=O)NCCSC(C(=O)N(CCCCCC)C(=O)CC)C)sccc1C#N Cc1ccc(C)c(C(=O)NC2CC(C)(CNC(=O)CC3CCCOC3)C2)c1 C12(C(=O)NCCCCN(C(COCC(=O)OC)=O)C)CCCN1CC(O)C2 c1(C(C(N)=O)NC(c2c(Br)noc2C)c2n(CCCC)nnn2)ccc(F)cc1 CCCC(C)(CCC)C(=O)NCC(C)CNC(c1cnn2c1OCC2)=O Cc1cc(C(=O)NC2CN(C(=O)C(c3cccnc3F)(C)C)C2)c(C)s1 C1(NC(C(C)OCC#C)=O)C2CC1CN(C(=O)C(N1CCC(C)C1)=O)C2 C1(N(C(c2ccc(SC)s2)=O)C)CN(C(c2ccc(F)cc2O)=O)CC12CC2 C1(CCNC(=O)OC(C)(C)C)(NC(CC2CC2(F)F)=O)CCCC1.C(=O)NC Cc1cnc(C(=O)NCCN(C(c2n[nH]c(C)c2F)=O)C(C)C)c(Br)c1 C=CCCCCCN=c1ccn2ncc(S(=O)(=O)NC(C)CC(C)C)c2[nH]1 C1(CC=C)(NC(c2nc(Cl)ccc2Cl)=O)CCCN(C(c2n[nH]cc2C)=O)C1 C(CO)(C(=O)N1CC(c2cc(C3COC3)[nH]n2)C1)NC(=O)OC(C)(C)C c1(C(=O)NCc2c(C(=O)NC(CCSC)CO)con2)cnn(C)c1Cl CC1(C)CCOC1CC(=O)NC1CN(C(c2cccnc2C(F)(F)F)=O)C1 C1(CNC(C2(C)CC2(F)Cl)=O)CN(C(c2ccc(CO)c(Cl)c2)=O)CCC1(F)F C(=O)(C1CSc2ccccc21)NC1C(NC(C=Cc2c(C)n(C)nc2)=O)COC1 C1(C(=O)OC(C)(C)C)(CNCc2cc(OC)n[nH]2)CCCC(=O)N1 N1(C(C(C)OC)=O)CC(CNC(=O)C=Cc2ccc(C(C)(C)C)cc2)CC1(C)C C1(NC(C#C)(C(=O)OC)C(F)(F)F)CCc2nc(C#N)sc2C1 c1(C(N2CCC(CNC(c3nc(C)sc3)=O)C2)=O)ccc(Cl)nc1C CCCCC(C(=O)NCC1CN(C(=O)CCN(C)CC)CCC12CCC2)C(C)C N1(CCNC(C(C)n2cccn2)=O)CCN(C(C2(C)C=CCCC2)=O)CC1 c1(OC)ccc(-c2nccn2CCC2CC2c2cnn(C)c2)cc1Cl N1(C(C2CC3(CC(CN=[N+]=[N-])C3)C2)=O)CCC2(CC1)CC(C1CC1)=NO2 c1(CC)cnc(CNC(=O)C(C)N(C(C2CCCCC2)=O)C2CC2)o1 c1(CC)cc(C)c(C(=O)NCCC(C)(C)CNC(=O)C(C2CCCCC2)F)o1 c1(C(=O)NCC(CC)(CC)NC(=O)C(O)C(C)OC)c(Cl)nc2ccccn12 c1(C(C)C(=O)NC2CC(C(F)C(=O)NCC(O)(C3CC3)C3CC3)C2)ccn(C)n1 N1(C(C(Cn2cccn2)NC(c2nn(CC)c(O)c2)=O)=O)CCC2(CCSC2)C1 N=c1c(C(=O)NCCCn2cc(CCOCCO)nn2)c[nH]c2ccc(Br)cc12 NC(=O)CC(O)C(=O)NCCOCC(=O)NC1CC2(C1)CC2C(N)=O C1(C(N2CC(CNC(C3(CC)CCOCC3)=O)C2)=O)CC12CC(F)(F)C2 N1(C(c2ccc(C)cc2F)C(=O)NCCC#N)CCCSc2ccc(F)cc21 C1(O)(C(N(C)CCN(C)C(C2CCC2C(C)(C)C)=O)=O)CCc2ccccc2C1 N1(C(Cn2cc(CC)nn2)=O)CC(NC(C2(COC)CC2)=O)CCC1C c1(NC(=O)NC(CCOC)(C)C)c(N)cccc1Br Cc1ccc(C(=O)Nc2cc(Cl)ccn2)cc1Cl c1(C(C2CCCCC2)C(=O)NC(C=CC(=O)OCC)C)ccccc1F c1(N(C(C)CC(C)NC(C2(c3ccc(F)cc3)CCC2)=O)C(C)=O)csc(=NC)[nH]1 CCC(C(=O)NCC(C)CN(C(=O)CCc1ccc(C)s1)C)OC Cc1ccc(C(=O)N(C)CC2COCCN2C(=O)CCCn2cccn2)cc1 CC(C(=O)N1CCC(CNC(=O)COCC2CCCC2)C1)S(N)(=O)=O N1(C(Cn2c(C)ncc2)=O)CC(NC(c2cc(C(F)F)cc(F)c2)=O)C(C#N)C1 C1(CCOC)(NC(C2CCC(C)(C)CC2)=O)CCN(C(C2CC2F)=O)CC1 C(CCCCCNC(c1ccc(Cl)cn1)=O)NC(c1c(COC)ncs1)=O C(c1ccc(F)cc1)=C(C)C(N1CC2CC1(CNC(=O)C1=CCCC1)C2)=O C1(CC(=O)NC(CC)C(=O)NC23CC(F)(C2)C3)CCOC1(C)C N1(C(CC2C(C)CCO2)C(=O)N(C)C)CCNC(=O)C(N)C1 N1(C(C(C)c2cccs2)=O)CC(NC(c2c[nH]cc2-c2cnn(C)c2)=O)C(F)C1 CC(C(=O)NCC1CC(C(=O)N(C2CCC2)C2CC2)C1)N1CCCC1 Cc1c(NC(c2ccc(Br)cn2)C)ncnc1N1CCC(C2CC2)C1 N1(C(c2c(C)oc(C(C)C)n2)=O)CCCN(C(c2cn(C3CC3)nc2C)=O)CC1 c1(SCC(=O)NC(C(C)NC(Cn2ncc(CC)c2)=O)C)ccc(C(C)C)cn1 C1(C(=O)NCC2CCCC(C)C2)CCOCC1(C)C.c12ccccc1C(=O)N2 N1(C(C(C)CO)=O)CCC2(CC1)CC2C(N1CCCN(C2CC2)CC1)=O C=C(C)CC(C(=O)NCC#CC(F)(F)F)NC(=O)CCCn1ccnn1 c1(C(N2CC3(CC(NC(C(C)(F)F)=O)C3)C2)=O)cc2cccnc2[nH]1 c1(NCC(=O)Nc2cn(C)nc2)ccc2c(c1)OCCO2 C(=O)(C(C)CCC(C)(C)C)NC(CNC(C1CCN(CC(C)C)C1)=O)C C1(NC(CC(CC)O)=O)CC1C1CCCN(C(C2(COC)CCCCC2)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(O)(CCNC(C2CC(OC)C2)=O)C1 O=C(CC1=Cc2ccccc2C1)NCCC1CCCN(C(=O)C(O)CC2CC2)C1 CCCC(CC)C(=O)N1CCC(N(C(C2CC2C2(C)COC2)=O)CC)CC1 c1(CC)ncncc1C(=O)NC1CC1CNC(c1ccc(CO)s1)=O CN1CCCC2C1CCN2C(=O)CC1CC2CCC1O2 N#Cc1ccc(C(N2CCCC(O)(CNC(c3ccc(F)s3)=O)C2)=O)c(O)c1 CC(CCC(=O)N1CCC(CF)C1)N(C)C.C1(C(=O)N)(CF)CC1 C1(NC(c2c(CC)nns2)=O)CN(C(C2CC(F)C2)=O)C2(CCOCC2)C1 c1(C(=O)NCC2CC(C)N(C(=O)Cc3nnc(O)s3)C2)c(F)ccc2[nH]ccc12 CC1(C)OCCC1C(N1CCSCC1C(=O)NC1C=CC(CO)C1)=O c1(C(=O)NCC2N(C(C=CCN(CC)CC)=O)CC2)nc(Cl)c(Cl)c(N)c1Cl C1(CCCNC(CC2CC(=C)C2)=O)CCN(C(=O)CC2(CSC)CC2)CC1 C1(CC(=O)NCC2CC(NC(C3(CC=C)CCCC3)=O)C2)CC(CC)=NO1 c1(CN(C(=O)NCCC2(CN)CC2(F)F)CC)cc(F)cc(F)c1 C12(C(=O)NCCCCCNC(C(CC=C)CC)=O)CC(CO)(C1)OC2(C)C c1(N(C)CC)ccc(C(=O)NCC(C)CN(C(=O)C(C)(C)OC(C)=O)C)cc1 c1(NCC2(C)CC(F)(F)C2)ccc(S(=O)(=O)NCC2CSCCS2)cc1Cl c1(C(N(CCCN(C)C(c2nc(C(C)(C)C)cs2)=O)C)=O)cc(Cl)nnc1Cl CC1CCCC(NC(=O)CCCNC(=O)C(F)n2ccnc2)C1 c1(C(=O)NCC23CC2CN(C(c2cnc(S)[nH]2)=O)C3)ccc2oc(O)nc2c1 C1(NC(=O)Cc2cn[nH]c2)CCC(C(=O)NCC2(Cl)CC2)C1 n1(CC)ccc(CC(=O)NC(C)(C)C(C)NC(=O)OC(C)(C)C)n1 C1(N(C(C2=C(C)CC2)=O)C)CCN(C(=O)CCc2cncs2)CC1C c1(C(C(=O)OC)NC(CCO)c2ccco2)cccc2cncn12 N1(C(C2(C)CC(=C)C2)=O)CC2CCCC2(NC(c2onc(OC)c2Br)=O)C1 N1(C(c2ccc(COC)[nH]2)=O)CC2ON=C(C)C2C1 C1(C(F)(F)F)(C(=O)NCC(C)CNC(=O)C(F)=C2CCCC2)CCOCC1 c1(OCC)cncc(C(=O)NCC2C3CC3CN2C(=O)C#CC(C)C)c1 C1(C(=O)NCC2C(NC(c3ccc(-c4ccccn4)s3)=O)C2)CCC(F)CC1 CC(C)CC(CNC(C1CC(O)C(F)C1)=O)C(=O)N1CC(=O)NC2(CC2)C1 c1(COC)ncccc1C(=O)NCCNC1CCN(C(=O)CCC(C)=O)C1 N1(C(c2ccnc(CC)n2)=O)CC2CCC(CNC(c3csnc3C)=O)(C2)C1 C1(CC(C(CC(=O)NCC)=O)=O)CCN(C(=O)C(C(=O)OC)OC)CC12CCC2 C(=O)(C1=CNS(=O)(=O)N=C1C)N(C1CC2CN(C(CCN(CCC)C)=O)C1C2)C CCCCC(CNC(c1cc(C)n(CCO)n1)=O)NC(C1CCCO1)=O CCC(CC)C(=O)NC1CC(C)(NC(c2ccnnc2O)=O)C1 c1(C(C(=O)NC)N(CCS(=O)(=O)NC)CC)cc2c(s1)=C(OC)N=CNC=2OC C(=O)(C1CCCc2c(O)cccc21)NCC1CC(C)N(C(=O)C2=C(Cl)CCC2)C1 c1(Nc2ncc(CCNC(c3ncccn3)=O)s2)ncc2[nH]ncc2n1 C(CCN=C(NCc1n[nH]c2c1CCCC2)NCc1ccns1)SC Cc1nn(C)cc1CCC(=O)Nc1cccc(CNC(c2ncncc2F)=O)c1 CCC(Cc1ccc(N)cc1)C(=O)NCC1CC(NC(c2cnncc2C)=O)C1 C(=O)(CCC(F)F)NC(C)CCCNC(C1(C)CC1C(F)(F)F)=O Cn1nc([N+](=O)[O-])cc1CNC(=O)NCC(=O)NCC1(C)CCC1 N1(C(C(C)OCC)=O)CCOC2(C1)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(C(CCC(N)=O)N)=O)Cc2ccc(CO)cc2C1.c12csc(n1)NC(=O)C2 c1(C(=O)NC(CNC(CSCC#C)=O)C)ccc(NS(=O)(=O)CCCC)cc1 Cc1cc(C(=O)NCCC(C)(C)NC(c2cn(C)nc2C(C)(F)F)=O)nnc1O N1(C(c2c(CNC(c3ncn(C)c(=O)c3)=O)cccc2)=O)CCSC2CCCC12 c1(OCC(=O)NC2C(NC(c3cnn(C4CCC4)c3)=O)CC2)ccc(F)cn1 c1(C(=O)NC2C(NC(C3(OC)CCOC3)=O)CC2)sc(C(F)(F)F)cc1C N1(C(c2c(C)csc2C)=O)CC(C(=O)NCCC(F)(F)Cl)C2(CC2)C1 C1(C(C)C)(C(=O)N(C2CCC3CC23)C)CCN(C(C2CCOCC2)=O)C1 N1(C(Cc2c(C)cccn2)=O)CC(CN(C)C(C2CC(O)C2(C)C)=O)C2(CC2)C1 N1(C(c2c(C)scn2)=O)CCCC2(CCN(C(=O)CC3CCC(=O)NC3=O)C2)C1 C12(C(=O)NCC3(O)CC(NC(c4cccc[n+]4[O-])=O)C3)CC3CC(C(=O)N1)C2C3 CC1Cc2ccccc2N(C(=O)C=Cc2ccc(SC)s2)C1 N1(c2cc(CC)ncn2)CCC(NC(C2CSC2)=O)C2(CCC2)C1 CC1CN(C(=O)CCc2nccn2C)C1C(=O)NCC(C1CCCCC1)O C1(CNC(C2ON=C(C)C2)=O)(CO)CC12CCN(C(c1sccc1F)=O)CC2 N1(C(C2CC(NC(C(C)(C)OCC)=O)C(O)C2)=O)CC(C2CCCCC2)C1 N1(C(CC(COC)C)=O)CC=C(C(=O)NC2C=CC(CO)C2)CC1 N1(S(CC)(=O)=O)CCOC2(CCCN(C(c3cc(Br)cc(F)c3C)=O)C2)C1 CCC(CC(=O)NC(C)C(=O)NCC(C)(F)F)OC C1(C(=O)NCC(N2CC3CCC3C2)=O)CC2C(C1)C2(F)F C1(C(=O)NCC2N(C(CCCOC)=O)CCC2C)CCc2nnc(C(C)C)n2C1 c1(C(C)(C)NC(=O)N(C2CCCCS2)Cc2ccccc2)cnn(C(F)(F)F)c1 c1(CNC)cn(CCCCCNC(C2CCC(F)C2)=O)nn1 C1(NC(c2n(C=C)nnc2)=O)CN(C(=O)CCN2CCNC(=O)C2)C2(CCC2)C1 Cc1ncc(C(=O)NC(C)CCCNC(C2(C(C)(F)F)CC2)=O)[nH]1 N1(C(c2c(OC)nc(C)cn2)=O)CCS(=N)(=O)C(C)(C)C1 N1(C(C=CCC)=O)CCC2(CC1)CN(c1ccnc(C(=O)OC)n1)CCO2 N#Cc1cnc(NC(=O)CC2CCN(C(C3(NC(N)=O)CC3)=O)CC2)cn1 N1(C(CCN(CCCO)C(=O)C2CC2)=O)CCC2CCC12 c1(C(N2CC3CN(C(=O)C=Cc4ccc(Br)cc4)C3C2)=O)cc(Cl)c(F)cc1F CCC(C)C(C(=O)N1CCCOC(CNC(c2cc(C)c(C)[nH]2)=O)C1)OC N1(C(c2c(CCC)n(C)nn2)=O)CC(NC(=O)CN2CCSCC2)C(C2CC2)C1 c1(OC)cnc(Cl)cc1C(=O)NCC(C)N(C(=O)CCC(F)(F)F)C CC#CCCC(=O)NC1(C)CC(NC(=O)CC2CCN(C(C)C)CC2)C1 CC(O)C(F)(F)C(=O)N1CC(CNC(=O)CCC(C)(C)F)C(C)C1 CCC(C(=O)N1CCCC1CNC(=O)C(C)=C1CCC1)SC N1(C(CC(C)(C)SC)=O)CC2CC(C1)N2C(C1CC1C(F)F)=O c1(C(N2CCC(C)C(N(C(=O)Cc3cncnc3)C)C2)=O)cc(F)c(O)c(F)c1 c1(C(N(CC(O)CF)CC)=O)ccc(CNC(C2CC(=O)N(C)C2)=O)cn1 Cn1ccc2nc(N(C3CC(N)C3)Cc3cccc(Br)n3)ncc12 C1(CC(=O)NC(C)(C)C)COC2(C1)CN(C(=O)CCNC(=O)CO)C2 n1(CCCOC)[nH]cnc1=NC(=O)C(C)N1CCCC1 N1(C(c2nc(C)n(C)n2)=O)CC2(CCN(C(C3CC3CF)=O)CC2)C1C(C)C C(=O)(C1=CS(=O)(=O)CCC1)N1C(C)CCC(NC(=O)C=Cc2ccc[nH]2)C1 C1(NC(c2cn(CCCOC)nc2)=O)CC(NC(=O)CO)C12CCOCC2 N1(C(c2cc(C)cc(O)n2)=O)C2CCC1CC(CNC(=O)CC13CCCC1C3)C2 CCC(C)(C(=O)NCC1(O)CN(C(=O)C(c2ccccc2)F)C1)C(F)F N1(C(C(c2ccccc2)C)=O)CCCCCC(NC(c2cc[nH]n2)=O)C1 c1(C(C(=O)NC2CC(COCCCC)C2)C)cccc(OC(C2C(C)C2)=O)c1 N1(C(C(C)Sc2ccc(C)cc2)=O)CC2=C(C1)CN(C(c1coc(C)n1)=O)C2 c1(C(N2CCN(C(CC(=O)OC)=O)CC2)=O)ccc(F)c(SC)c1 C1(NC(C2CCC(CC)O2)=O)CCC2(CC1)CCN(C(=O)COCCC(C)C)C2 CC1=C(C(=O)NC2CCN(C(c3ccncc3N)=O)C2)Cn2nnnc2N1C Cc1noc(C)c1C(=O)NCC1C=CCN1C(=O)COCC(F)(F)F C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)(C(C)C)NC(c1cncc(C)c1)=O c1(CN2CCC(C)(C(N3CCS(=O)CC3)=O)C2)cc([N+](=O)[O-])ccc1Br c1(SC)ccc(C(N2CCCC2CNC(c2ccc(C3CCC3)cc2)=O)=O)cn1 CN1Cc2ccc(C(N3CCC(CNC(c4ncc[nH]4)=O)C3(C)C)=O)cc2C1 C12(C(N3CCC(OCCNC(c4cc(C)[nH]n4)=O)CC3)=O)CC1COC21CCC1 C1(C(=O)NCC2(NC(C3CCCN(C(=O)OC)C3)=O)CC2)C2CCC3C(C2)CC13 N1(C(Cc2cccc(C)c2)=O)CCC2(CCC(NC(c3ccc(Cl)s3)=O)C2)C1 Cc1ccn(C(C)C(=O)N(C(C)CN(C(=O)CN(C)C(N)=O)C)C)n1 c1(-c2nc(NC(CCC(CC)NC)=O)sc2)ccc(C(C)(C)C)cc1[N+](=O)[O-] c1(N2CCCC(C(N(C)CC3CCNC3)=O)C2)ncc2nccnc2n1 Cc1cc(C(N2CCOC(C)(CNC(=O)CN=S(C)(C)=O)C2)=O)c2n[nH]cc2c1 CCC(CC)CCC(=O)OCC(=O)NC(c1cccc(Cl)c1)c1ccc(C)cc1 CCCCCS(=O)(=O)CC(=O)NC1CN(C(C2CCCN2C=O)=O)CC2(CC2)C1 c1(C(=O)NCC2OCCN(C(C(CC)F)=O)C2)cc2c(nc1O)CCC(C)(C)C2 C1(C(=O)NC(C(O)CO)C2CC2)CC(O)CN1C(=O)CCc1cncnc1 N1(C(C(C2CCN(C(C(C)C(=O)OCCF)=O)CC2)C)=O)CCC(C)(C2CC2)C1 C1(CNC(C2CCN(C(C3(c4ccncc4)CCC3)=O)C2)=O)CCCC2CC12 c1(C(N2CCC(C(CO)NC(C3C4CC5C(C4)C35)=O)CC2)=O)cc2scnc2[nH]1 c1(OC)cccc(NC2(C)CC(NC(c3cccc4c3ncn4C)=O)C2)c1[N+](=O)[O-] C1(NC(C2(OCC)CCCC2)=O)CC(C(=O)NCC2(C#N)CCC2)C12CCC2 C(CCCC(=O)N1CCCC1CCNC(=O)C(C)CCN(C)C)SC c1(C(=O)NCC(CNC(c2c(CCC)nco2)=O)O)cncc(OC(C)C)c1 N1(C(C=CCCC)=O)C2CCCC1CN(C(c1cccc(=S)n1O)=O)CC2 c1(N(CCC)CC)ccc(C(=O)NC2(F)CCN(C(=O)NCC=C(C)C)C2)cn1 C(=O)(CC(=O)NCC(C)N(C)C(c1cnn(C2CC2)c1)=O)NCC c1(NCC(=O)NN2CCC(N(C)CC)CC2)ccc(S(=O)(=O)NC2CNC2)cc1 C(=O)(C1=CCCCN1C(=O)OC(C)(C)C)NCC1(C)CC(NC(C)=O)C1 c1(C(C)NC(C)(CCn2cccn2)c2cccs2)ccc2c(C)[nH]nc2c1 C(C1=CCN(C(=O)C(c2ccccn2)O)CC1)NC(C=C(C)Cl)=O C(=O)(C(O)P(C)(C)=O)NC1C2CN(C(c3cc(OC(C)C)ncc3)=O)CC21 c1(C(C(=O)N)C)ccc(C)cc1.C1(CC(=O)OC)(CCCN(C(C)=O)C)CCCC1 N1(C(COCCCOC)=O)CC2CC2C1C(=O)NCC1(C)CC(C)(C)C1 C1(NC(C2CCCN(C(C(CO)OC)=O)C2)=O)CC12CCOCC2 C1(NC(C2CCN(C(C)=O)CC2)CC)CCCC(C)(C)C1 C#CC1(CN2C(CC(C)N(C(=O)NC(C)(C)C)CCO)CC2)CCOCC1 CC(CSc1ccccc1)C(=O)N1CC(=C2CC(NC(=O)Cc3cocn3)C2)C1 N1(C(c2c(C)nc[nH]2)=O)CC2(CCCN2C(=O)CCc2ccccn2)C1 C1(C(N2CCCC(C)C2CO)=O)(OC)CCN(C(=O)CCc2nccs2)CC1 Cc1cc(C(=O)NC2CC2NC(c2nocc2C(C)C)=O)sn1 C1(C(=O)NCC(COCC)F)CC(NC(=O)CCC2CC(CSC)C2)CCO1 c1(C(C(=O)NCCOCC)N(C(C)CCC(C)C)C)nn(C)nc1Br c1(CC(=O)NCCN2CCC(NC3CCC4(C3)N=N4)CC2)c(Cl)cccc1Cl C1(C(N2CCCC2)=O)CC2(C1)CC21CC1.C(CC(C)C)(C(=O)NCC1CC1)NC(C)=O C12(C(=O)NCC3(O)CN(Cc4nc(C)c(C)o4)C3)CCC(CF)(C1)OC2 CCCC(CCC)C(=O)N1CCN(CC(=O)NC2(CO)CC(F)C2)C(=O)C1 C1(C(=O)NCC(CCNC(c2cc(OC)ncc2)=O)O)Cc2cc(Cl)ccc2O1 c1(OC)cccc(CC2(CC(C)C)CCCN2C(c2cnc(Cl)cc2I)=O)c1 c1(CC)ccc(F)c(C(=O)NCC2(C)CCN(C(c3nc(C4CC4)cs3)=O)C2)c1 Cn1ncc(C#N)c1NC(C1CC(O)CCN1C(c1ccc(Cl)cc1F)=O)=O N1(C(COC2(C)CCCC2)=O)CCC2(CC(NC(=O)C(C)(C)CCCO)C2)C1 c1(CN2CC(C)(CC(=O)Nc3c(C(=O)OC)ccs3)C2)nc(Cl)ccc1F c1(NCCN(CC)CC)cc(=NC(C)c2ccc(O)nc2)[nH]c(C)n1 c1(Cn2cc(-c3ccc(OC)cc3OC)nn2)cn2cc(Cl)cc(Cl)c2n1 N1(C(C2C(CNC(c3ccc(O)nc3)=O)CC2)=O)CCC2CCCC2CC1 N1(CC(N2CC(CC(F)C(=O)NCc3ccc(O)cc3)C2)=O)C(=O)CCCC1=O CC1(C)CC(c2ccc(F)cc2)(C(=O)NC2CN(C(=O)C(C)(C)C3CCC3)C2)C1 c1(C(N(C)CC2(O)CN(C(C34CCCC3C4)=O)C2)=O)cc(Br)cnc1O c1(OC(CC(C)N(C)C)=O)ccc(Cl)cc1Br.c12ccccc1OCC2 C12(CNC(C(N3C(C(=O)OC(C)C)CCCC3)=O)=O)CCC(C(F)F)(CC1)C2 C=CC(C)(O)CC(=O)N1CCOC(CN(C(=O)CCc2ccc(C)c(C)c2)C)C1 C1(CC(=O)NCC(C(C)C)C)COCCN1C(c1ccc(CO)nc1)=O C(CC(=O)NCC1(F)CCOCC1)(C(F)(F)F)NC(C(COC)C)=O C#Cc1ccccc1CC(=O)NC(C)(C)CCN(C(=O)CCCC#CC)C CC(C(=O)NCC1(NC(C2CSC2)=O)CCOC1)C(=O)N1CCOCC1 C1(NC(c2cc(CNC(C3CCCC3)=O)oc2)=O)CC2CC1OC(=O)N2 CC(O)C(C)(C)CNC(=O)CC1(C)CCN1C(C1CC2CCC2C1)=O Cc1ccc(Cl)cc1C(N1CC(C)(NC(C2(c3cccnc3)CCCC2)=O)C1)=O C1(NC(c2csc(Cl)c2)=O)CCOCC1NC(C1CC(F)(F)C1)=O c1(CNC(C2C(C)CCCC2)=O)ccc(C#N)cc1F.C12CC(C)(C)CN1C2=O N1(C(CNS(C)(=O)=O)=O)CC2ON=C(CNC(c3ccc(CO)cn3)=O)C2C1 c1(CC(=O)NCC2(O)CN(C(CNC=O)=O)C2)ccc2nc[nH]c2c1 C(=O)(C1c2ccccc2C2CC1C2)N1CC(C)CC(NC(C(CC=C)CC)=O)C1 C(=O)(C1(C)CCCc2ccccc21)N(C1CC2CCCC(C1)N2C(=O)C1CC1)C c1(CN(C(C)C)C(=O)NCc2cccc(N)c2F)ccc(F)cc1F C1(NC(CNS(N)(=O)=O)=O)COC2(C1)CN(C(c1cc(CO)on1)=O)C2 C1(NC(=O)NC2(c3cccc(Cl)c3)CCC2)CC2C(C1)C2(F)F C1(=CC(N2CC(NC(Cc3cccc(C)c3)=O)C2)=O)C2CC3CC(C2)CC1C3 CC1CCN(C(C2CCSC2)=O)CCN1C(c1ccc(CO)c(F)c1)=O C1(NC(C=C(COC)C)=O)CC2C1CCN2C(c1nnn(-c2ccccc2)n1)=O Cc1cc(C(=O)NCC2CCN(C(=O)CCC3CC3(F)F)C(C)C2)cc(N)c1O N1(C(c2c(N)c(Br)ccc2)=O)CCC2CN(C(c3ccccc3)=O)CC12 CC1C2CCCCC2CN1C(C1CC12CCN(C(=O)Cc1cn(C)cn1)C2)=O C1(NC(=O)C=CCF)CCC(CCNC(c2cc(CCO)on2)=O)C1 c1(C(=O)NCC(CNC(CCc2nc(C)sc2)=O)C)nccc2c1NCCC2 C(CC1=CCCCCC1)NC1C2CN(C(C3N(CC)C(=O)CC3)=O)CC21 C1(C(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)CCc2ccccc2)C1 c1(C(=O)NC2CN(C(C(=CC3CCCC3)C)=O)C2)ccc(Br)cc1O C12CCCC3CN(CC13)C(=O)N2.CC(CCC1CCCO1)NC(=O)OC(C)(C)C c1(CCC(=O)NCCN(C(=O)CN2CCCNC2=O)CCC)cncc(F)c1 c1(C(=O)NCc2c(C)nn(C)c2)ncn2cc(-c3ccncc3F)sc12 CCC(C(=O)NC1CC(NC(c2c(Br)ccc(F)c2F)=O)C1)C(C)(F)F C(=O)(C(CC(C)(F)F)NC(=O)OC(C)(C)C)NCCCNC(CCC(C)F)=O N1(C(CCC(=C)Cl)=O)CCCC(NC(=O)C(C(C)C)n2cnc(C)c2)CC1 c1(C(=O)NC(C2CCCN(C(=O)Cc3cncn3C)C2)C)cc(N)ccc1F c1nc2cc(F)c(F)cc2[nH]1.N1(Cc2nnn(C)n2)C(=O)CN(C)C1=O Cc1ccccc1C(C)C(=O)NCC1COCCN1C(C1CC1F)=O Cc1nncc(C(=O)N(CC(=O)NCC2Cc3nccn3C2)C2CCC2)c1C C1(C(N(C2CN(C(=O)C(F)=C3CCC3)C2)C)=O)CCC(=O)N2CCCC12 C1(CNC(C(CCC)CC)=O)CN(C(=O)Cc2cccn2C)CCC1(F)F Cc1cc(-c2cn(CC3CCCN3C(=O)CCOC(C)C)nn2)sc1C N1(C(CNC(=O)OC)=O)CCC2(CCC(NC(=O)COC3CCCCC3)CC2)C1 Cc1nnn(C)c1C(=O)NCC(C)NC(=O)CCCc1cccs1 CC1(C)CCC(=O)N(NC(=O)C2(Cl)CC2C(=O)OC(F)F)C1=O c1(OCCC)ccccc1C(=O)N(CC(O)CN(C(=O)C(C)(C)C#N)C)C c1(-n2c(-c3c(C)onc3)nc(Cc3cccc(Br)c3)n2)cc(Cl)ccc1C(F)F c1(C(=O)NCC2(C)OCCN(C(Cc3cn(C)nc3)=O)C2)cnc2[nH]nnc2c1 CC1=C(C(=O)NCC2CCCN(C(=O)CCc3ccoc3)C2)CCCC1 C=CCC(C(=O)NCCCOc1ccc(C(O)CF)cc1)c1ccccc1 C1(C(=O)OC)(COC)CN(N2CCOC(C(N)=O)CC2)C1 C1(C(=O)NCCc2nccs2)CCC2(CN(C(c3cc(F)c(Cl)c(Cl)c3)=O)C2)O1 c1(C(=O)NCC2C(NC(c3c(C)cc(C(F)F)o3)=O)COC2)c(C)cc[nH]c1=N CC(C)(C)C#CC(=O)N1CC(CNC(c2ccc(NC3CC3)nc2)=O)C(O)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(CC(C)NC(C(C(CC)C)OC)=O)C1 Cc1ccc(C(c2nnnn2C2CCC2)NC2CC(C)(C)CCC2O)c(C)c1C N1(C(CCc2ccc(C)s2)=O)CCCC12CCCN(C(=O)C(C)c1cc[nH]n1)C2 Cc1cc(C#N)ccc1NCc1cnn(-c2ncccn2)c1C N#Cc1ccc(C(=O)NC2CCCN(C(=O)CC3(C(F)F)CC3)C2)cc1F c1(C(=O)NCC2CN(C(CC=CCC)=O)C(C)C2)cn(C)c2ncccc12 c1(C(=O)NCC2CC(NC(Cc3ccc(OC)cn3)=O)C2)cc2ncccc2o1 CC1(CCNC(C2(F)CC2)=O)CCN(C(c2cccc(O)c2F)=O)CC1 C1(CC)C(NC(c2sc(C)nc2C)=O)CCN1C(=O)C(CO)NC(=O)C(C)C Cc1ccc(F)cc1CN1CCN(C(c2ccccc2Br)C(=O)NC2CC2)CC1 c1(C(=O)NCC2CC(NC(C(C)NS(C)(=O)=O)=O)C2)c[nH]nc1C(F)F c1(C(=O)NC2CCN(Cc3onc(COC)n3)CC2C)c(C)sc2ccccc12 c12ccccc1NC(=O)N1CC(CC)(C1)C2.c1(C(C(C)C)OC)ccc(Cl)cc1 N1(C(c2oc(C)c(CO)c2)=O)C2CCC1CC(CNC(C1(C)CC(F)C1)=O)C2 C1(C(=O)NCCN(C(C(C)OCC2CC2)=O)CC(F)(F)F)CCC(N(C)C)CC1 Cc1nc(Cl)[nH]c(=NCC2CN(C(=O)COCC3CCOC3)CCCO2)c1F C1(C(N2CCC(CNC(=O)CC3OCCCO3)C2)=O)(OC)CC(CF)C1 c1(NC2C(CC=C)CCCC2)nccc(=NC(C)c2nc(C)cs2)[nH]1 c1(C(C)(C)C)cc(C(=O)NCCC2(NC(C3(C)CCCO3)=O)CC2)no1 N1(C(c2nc(OCC)sn2)=O)CCC(N(C(C2(CC(F)F)CCC2)=O)CC)CC1 C=CCC(CNC(c1ccc(OC)nc1)=O)C(=O)NCCCN1CC=CC1 C1(C(=O)NC2CCC(CNC(C3(OC)CCOCC3)=O)C2)COC2(CCC2)CO1 C12(CNC(CC(CC=C)(C)C)=O)CCCCC1CN(C(=O)CN(C)CC)C2 C1(NC(c2c(CC)ocn2)=O)CN(C(C2(C)COC(=O)C2)=O)Cc2ccnn2C1 c1(CC(=O)Nc2ccc(-c3ccc(F)cc3)nn2)ccnc(Br)c1 c1(C(=O)NC(c2cccs2)(C)C)coc(CNC(c2nc(Cl)cs2)=O)n1 C(=O)(C(F)C(C)(C)O)N1CC2C(CNC(c3c(C)oc(C4CC4)n3)=O)(C2)C1 c1(C(N2CC(CCO)(NC(CCCOC)=O)C2)=O)cccc2c1NCC(C)C2 Cc1nc(O)sc1C(=O)N(C1CN(C(=O)C(C)C(C)C)C1)C C(=O)(C1Cc2ccccc21)NCC(C(=O)NC1CCN(C(=O)CCF)C1)O C1(C(N(CCOC)CC)=O)CCCCCN1C(c1cnncc1OC)=O C1(CNC(C2CC(C(C)C)OC2)=O)CCN(c2nc(C(=O)C(C)C)ns2)C1(C)C N1(C(C(C)(C)C2CCN(C(C3CCCC(=O)N3)=O)C2)=O)CCCC2(CC2)C1 c1(CNC(COCCNC(CSC)=O)=O)ccc(C)c(O)c1 C1(CNC(C(C=C=C)C)=O)CN(C(c2ccn(CC)c2C)=O)CCC1(F)F C1(NC(=O)C=Cc2ncc[nH]2)CC2CCC(C1)N2C(c1ccc(F)c(Cl)c1)=O N1(C(C2CC(=C)C2)=O)CCC(N=c2cc(C)[nH]c(C(=O)OC)n2)C(C)C1 C(=O)(Nn1ccccc1=O)C1(CNC(C2CC(C)OC2C)=O)CC2(CC2)C1 C1(C(=O)NCCN(C(C2(Cl)C(C)(C)C2)=O)C2CC2)CC1C1CCCC1 c1(CC(=O)NC2C(NC(C(CNC(C)=O)(C)C)=O)C2)ccc2c(c1)OC(F)(F)O2 C(=O)(C1=CC2C=CC(C1)C2)NCCNC(CC(COC)C)=O N=c1[nH]cnc2c(C(N3CCC(CNC(=O)C(O)C4CC4)C3)=O)cnn12 c1(CC(=O)NC(C2(O)CN(C(C(CCCC)O)=O)C2)C)ccc2c(c1)CCCS2 N1(C(C(CCSC)NC=O)=O)C2CCC1CC(NC(=O)CCP(C)(C)=O)C2 C1(NC(CC2N(C)CC=CC2)=O)CN(C(=O)CCCF)CC12CC2 C(CCC(O)C(=O)NC1CCC(SCC)CC1)NC(Cn1c(CCC)ncc1)=O C(=O)(C(CO)C(C)(C)C)N1CCC(NC(COCCCCCC)=O)C1 C(C(C(=O)N1CCC1C(N)=O)C(C)(C)C)NC(c1cnc(C)o1)=O C1(CC)(NC(c2cnc(OC(C)C)cn2)=O)CCCN(C(c2occc2C)=O)C1 CC1(C)CN(C(c2cccc(Br)c2F)=O)CC1NC(c1ccncc1N)=O C(=O)(C(C)(C)C(=O)NC1(CNC(C2(OC)CCSC2)=O)CCCCC1)OC CC1(C)CN(C(C2CC3CCC2O3)=O)CC1CNC(c1cc(CO)ccn1)=O c1(C(N(CCCCNC(=O)COC2CC=CC2)C)=O)ncccc1N(C)C C1(NC(Cc2nc(CC)sc2)=O)CCC(CC(N2CCC(CCO)CC2)=O)CC1 c1(CCC(=O)N(C)CCNC(C2(F)CC(C(=O)OC(C)(C)C)C2)=O)ncccc1F c1(NC(C2C=CC(NCc3cnc[nH]3)C2)=O)ccc(Br)nc1CO c1(CC(C)OC(C23CC(F)C2C3)=O)ccc(Br)cc1Cl CC(CC#C[Si](C)(C)C)(C(=O)O)NC1CCCc2c(O)cccc21 N1(C(C(C2CC2)OCC)=O)CCC2CN(C(C3(CO)CC=CCC3)=O)CC2C1 N(C1CCCc2ccc(F)cc21)Cc1n(C2(C)COCC3CCCN23)c(CO)nn1 CC1(C)C(CC(=O)O)CN1Cc1ccc(CCCN)cc1 Cc1cc(C(=O)NCC2CCN2C(=O)Cc2cccnc2C)c(O)nn1 C1(O)(CCNC(=O)Cc2nc[nH]n2)CCN(C(=O)CC2CC(=O)NC2=O)CC1 N1(C(c2ccn(CCCC)n2)=O)CC(C)N(C(=O)CCN2CCOCC2)CC1C C1(CNC(CN(C)C2CC2)=O)CN(C(=O)CC2(O)CCCCC2)CCCO1 c1(CC)ccnc(C(=O)NCC2CCN(C(=O)CC3CCCCC3O)C2)c1 N1(C(CC(=O)OCC)=O)CCN(C(c2cc3sc(CC)cc3s2)=O)CCC1C C1(C(=O)NC2CC3CN(C(C4(SC)CC4)=O)C2C3)Cc2ccccc2C1 C#CCC(C)C(=O)NCC1CCC(CNC(=O)Cc2ccc(CO)cc2)CC1 c1(C(=O)NC2C3N(C(CC(CCC)C)=O)C(CC3)C2)cc2ccccn2c1 c1(OC)ccc2c(c1)N(C(=O)CCCCC(C)(C)C)CCN2 c1(C(=O)NC(C)C(C)(C)NC(=O)C(O)C(F)F)ccc2c(c1)CCCC(=O)N2 c1(OC)ccc2ccccc2c1CN1CCC1C(=O)NCc1cn[nH]c1 C(C1Cc2ccccc21)NC(=NCCC#C)NC1CC1C1CCCCC1 C(=O)(C(CCNC(c1cc(CC)oc1C)=O)OC)NC(C1CCCO1)CC N1(c2c[nH]c(=N)s2)CCC(C(=O)OCC2CCCC2)CC1 CCCCC(C)C(=O)NCCC1(CNC(C2CCC(N(C)C)C2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)NC1CCC(CNC(=O)CC2CCNC2=O)C1 Cc1[nH]nc2c(C(N3CCCC(NC(=O)C(C)N4CC(C)C4)C3C)=O)cccc12 C1(C(F)(F)F)CC(N=c2[nH]c(NCCC34CCCN3CCC4)nc3c2CSC3)C1 C1(N2CC2)(NC(C(CC(C)C)ONC(c2csc(C)c2C)=O)=O)CCC(C)(C)C1 N1(C(C23N(C(=O)OC(C)(C)C)C(CC2)CC3)=O)CC(C2CCCCC2)C1 c1(N2C3CC(=O)NCC2CC3)nc(=NCCc2ncccc2F)[nH]c2c1COC2 C=CCC(C)(CNC(=O)C(C1CC1)NC(=O)C(F)C1CCC1)CO N1(C(CCc2cc(C)on2)=O)CCC(N(CC(C)C)C(C2CC2C)=O)CC1 N1(C(C2(CC#C)CCOC2)=O)CCCCC(CNC(=O)CC2CC(C)OC2C)C1 C(=O)(CC(C)CN(C)C)N(CCOC)CCNC(C1(C)CC1C(F)(F)F)=O N1(C(COCCOCC)=O)CC(N(C)C(C2CC3CCC2CC3)=O)C(C)(C)C1 C1(C(N2CC(CNC(CN(CCCCCC)C)=O)C2)=O)CC(C(C)=NO)C1(C)C C1(C)(CNC(c2c[nH]c(=NC)s2)=O)CN(C(C2(C)C=CCCC2)=O)CC1C Cc1nc(N2CC(C)CC(C)C2)c2cnn(CC#N)c2n1 C1(CC(N)=O)(NC(c2ccc(SC)s2)=O)CCN(C(c2nc(C)ccc2C)=O)CC1 c1(C(N2C(=O)NC(CC(C)C)C2=O)C)ccccc1[N+](=O)[O-] c1(C(=O)NCC2(C)CCCN(C(=O)CO)C2)nnn2c1CCCC2 c1(C(N2CC(NC(c3sccc3Cl)=O)C(O)C2)=O)cc(F)c(F)cc1Cl C1(CNC(=O)OC(C)(C)C)CCCCC1C1CC1.C1(NC(=O)N)CC(CO)C1 N1(C(CN(C)C)=O)CCCC2(C1)CN(C(c1cc[nH]c1)=O)C2.c12ccccc1S2 c1(C(=O)NCCNC(C(=O)N(CCCOC)C)=O)cc(Cl)c(OC)c(Cl)n1 c1(C(N2CCC(N(C(=O)CCn3cnnn3)C)CC2)=O)cc(F)c(CO)c(F)c1 N1(C(c2sc(C)c(O)n2)=O)CC(NC(=O)C(O)C2CCCC2)C2CCCC12 N1(C(c2cccc(CC=C)c2)=O)CC2CCN(C(c3cc(C)c(Cl)s3)=O)C2C1 Cn1cc2c(n1)CCCC2C(=O)NCC1(C)CCN(C(c2ncc(F)cn2)=O)C1 C(C(F)(C(=O)NC(C)(C)CC(=O)OC)C(C)C)NC(C(COC)NC(C)=O)=O c1(C(=O)NC(C(C(C)C)NC(C(C)=C(C)C)=O)C)cccc2ncsc12 N1(C(C2C(C)(C)C2NC(C2CCNC(=O)C2)=O)=O)CCCCCCC1CO N1(C(C(CC)OC)=O)CCCC(C2(NC(C3COC4COCC34)=O)CC2)C1 C1(CC)CCCCCCN1C(=O)CNC(C1CC(=O)C12CCC2)=O N1(C(CCC#CC)=O)CCCOC(CNC(=O)C(F)C2CCC2)C1 N1(C(CCCOCC)=O)CC(CC)CC1CNC(=O)C(CC)N(C)C C1(CC(=O)N(C2CCN(C(c3cnc(Cl)s3)=O)CC2)CC)CCCS1(=O)=O C(=O)(C(CC)CC=C)NCC(C#C)OC.C1(=O)CCCN1C CCC(C(C)C)NC(=O)C#CCNC(c1cnc(C)o1)=O C1(N(CCOC)C(C2(C)CC2C(=O)O)=O)CCNCC1 C1(C(=O)OCC)CCCCN1C(C1CCN(c2cnn(C)c2)C1=O)=O C(=O)(C1=C(C)CCOC1)N1C(C(N(CCCCCC=C)C)=O)CC(C)(C)CC1 CCCCCC(C)(C)C(=O)N(CC(=O)NC(c1cnn(C)c1)CO)C1CC1 CCC(CC(=O)NCC(CNC(=O)Cn1cc(Cl)c(C)n1)S(C)(=O)=O)C(C)(C)C c1(C(=O)OC)ccnnc1O.C1C(CC2CC2)C(=O)N1C(C)C(=O)N1CCCC1 Cc1ccc(CCC(=O)NC(CNC(C2CCO2)=O)Cc2ccc(F)cc2)cn1 C(CCCCN(C(=O)CC1CN(C)C1)C)NC(C(C)SC(C)C)=O c1(C(N2CCC(C(C)(C)NC(c3[nH]n(C)c(=O)n3)=O)CC2)=O)ccc(O)c(Cl)n1 N1(C(C2(COC)COC2)=O)CCC(C)C(NC(c2ccncc2SC)=O)C1 C1(CC=C)(NC(c2cc(-c3ccns3)on2)=O)CN(C(c2ccoc2Br)=O)C1 C12(C(N3CC(C)CC(NC(C4=C(C)CCC4)=O)C3)=O)CC3CC(C1)CC(C)(C3)C2 c1(C2(C(=O)Nc3nccc(CN)c3)CCCC2)cccc(F)c1F Cc1cc(NC(=O)C2CC2)ncc1-c1nc(C2CCC3CC3CC2)no1 N1(C(CNS(NC)(=O)=O)=O)CC2CCC1CN2C(=O)CCOc1ccccn1 C1(NC(c2ccc(CO)s2)=O)CC(=O)N(C2CN(C(c3ccc(CO)s3)=O)C2)C1 c1(C(=O)NC(CCOC)C(=O)NCCc2cnc(C)[nH]2)c(C)cccc1O N1(C(=O)NC(c2ncc(C)[nH]2)C)CCOc2ncccc2C1 c1(C(N2CCN(CC3CCN(C(C)=O)CC3)CC2)=O)cc(I)c(Cl)cc1Cl Cc1ccc(C)c(OCC(N2CC(C(=O)O)CC2C)=O)c1 C1(NC(c2cccnn2)=O)CN(C(c2snc(O)c2Cl)=O)CC2(CC2)C1 C1(C(=O)NC2C(CNC(c3cc(CC(C)C)[nH]n3)=O)CC2)CN(S(N)(=O)=O)C1 c1(OC)ccccc1C1CN(Cc2nonc2C)CCO1 c1(C(C)Nc2c[nH]c(-c3ccc(C(F)(F)F)cc3F)c2)cccc(Cl)c1Cl c1(C(N2CCOCC(NC(C3CC34CCCC4)=O)C2)=O)cc(Cl)cc(F)c1F c1(SC)c(C(=O)NC(C)C(CO)NC(=O)Cc2csc(C)n2)cnn1C C(CCCCC(=O)NCc1c[nH]nc1C(=O)NC1COCCC1(F)F)OCC CC1OCCC1CC(=O)NCCOC(C)(C)CNC(c1nocc1C1CC1)=O c1(OC)ccc2c(c1)CCCC2NC(c1ccn(CCF)n1)=O C1(NC(c2cc(C)c(=O)n(C)c2)=O)CCC2(CC1)CC(NC(C1CC1CC)=O)C2 N1(C(C)C)CC2CC1CN2C(=O)CONC(C1CCOC(C)(C)C1)=O c1(CC(=O)NC(CC(C)NC(c2cn(C)[nH]c2=N)=O)C)cc(Cl)cc(Cl)c1 N1(C(CCCNC(C)=O)=O)C2CCC1CN(C(C1COCC1C(F)F)=O)C2 C1(COC(c2csc(-c3cnn(CCO)c3)n2)=O)CCCOC1 n1(CC(=O)NC(C)CC2CN(C(=O)CC3CCC3)C2)cnc(Br)c1 C1(NC(CC2(NC(c3cnn(C)n3)=O)CC2)=O)CC12CCCCCC2 C#CCCCCC(=O)N1CC(NC(=O)CCc2nnc(-c3ccsc3)o2)CC1C CCCC(C(=O)N1CCC(NC(c2cccc(C(C)(F)F)c2)=O)CC1)NC(N)=O C=C1CCN(C(=O)CN2CCC(OC)C2)C(C(N2CCC2CO)=O)C1 C1(NC(CCCCC=C)=O)CCN(C)C12CCCN(C(=O)C=CC(=O)N(C)C)C2 CC1(F)CCN(c2nnc(-c3cccc(OCC(F)F)c3)n2CC(N)=O)C1 c1(N)ccc2nccn2c1.n1(C(CC)(C)C)nnnc1C1C(COC)C12CC2.CC n12cc(nn1)C2.n1(C2(COCC)CCC2)cc(C)cn1.C(=O)(CCOCCO)NC C1(CNC(c2cncc(Cl)n2)=O)CC2CN(C(=O)CSC3CC3)CC12 O=C(C1=CCSC1)NCC1(C(=O)NCc2nn[nH]c2C2CC2)CCCO1 c1(SCC(=O)NCC2(NC(=O)C=C(Cl)Cl)CCOC2)nccc2ccccc12 c1(N(C(c2ccnc(CO)n2)=O)C(C2CCCNC2)C2CC2)cccc2c[nH]nc12 N1(C(Cc2c(C)noc2C)=O)CCCC(C)C1CCNC(C1(C(C)C)CC1)=O CCCCC(O)C(=O)NC1C2CC1N(C(C1CN(C3CCOCC3)C1)=O)C2 c1(C(=O)OC)cc(C(=O)OOC)oc1C.N1(C(CC)=O)CCC(C)C1 CCCC(O)C(=O)N1CCC(CNC(c2ccc(-c3nnc(O)o3)cc2)=O)C1 CC1OC2(C(=O)NC3CN(C(=O)Cc4cnccn4)CC3C)CCC1CC2 C(CC(C)(C)CC(=O)N(C)CCOc1[nH]nc(C(F)(F)F)c1C#N)OC c1(C(=O)NCCN(C(C2C(C)(C(=O)OC)C2)=O)CC2CC2)ccc(OC)c(OC)c1 CCCCCCC(CC)C(=O)NCC1CCN1C(C12CCC(CC1)C(C)O2)=O C1(NC(C(N2CCC(O)CC2)C)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1F C1(OC)CC(CNC(C2(C(=O)Nc3cccc(Cl)c3)CC2)=O)N(C(=O)CO)C1 C1(OC)CCN(C(C2(F)CCN(C(c3cncc(C)n3)=O)CC2)=O)C12CCC2 c1(CNC(C2CSCN2C(=O)CC2CCCC2)=O)ccncc1Cl C=CCCCC(C)(C)C(=O)N1CC2CC2(C(=O)Nc2ccccc2C(C)(C)C)C1 CC1=C(C(=O)NCC2CC(C)CN(C(=O)CCC3CCCO3)C2)CCC1 C1(CC=C)(C(=O)NCC(N)=O)CCCN1C(=O)CC1CCCCO1 c1(OCC)ccccc1C(=O)N(CCC(C)NC(=O)C(=O)NCCC(N)=O)C c1(C(=O)NCC(CC)NC(=O)CCF)cc(OC)c(Cl)cc1Cl CCC(C)(C(=O)NC1CC2CCC(C1)N2C(=O)C=CC(C)C)C(F)F c1(NC(=O)CC2(c3ccccc3)CCCO2)cccc2c1OCC2 C1(NC(=O)CCCc2cccs2)CN(C(c2cnns2)=O)CCC1CO c1(C(C(=O)NCC(C)N(C(=O)Cn2cccn2)C)OC)ccccc1C(F)(F)F c1(OCC)nc(C(=O)NC2(CNC(C3(C)CC3(C)C)=O)CCC2)co1 CC1CC(C(=O)NCC2CCN(C(C3(C(N)=O)CC3)=O)CC2O)CC(=O)N1 C1(CNC(C=NOC)=O)CCC2CN(C(C3CCC(C(N)=O)C3)=O)CCC2C1 N1(C(CCC=C)=O)CCC(CNC(=O)Cc2ccnc(F)c2)C(C)(C)C1 c1(C(N2C(CN(C)C(C3CCCC(O)C3)=O)CCC2)=O)cc(N)cc(O)c1F c1(CC(=O)NC2C(CNC(C3(COC)CCCO3)=O)C2)cccc(OC(F)F)n1 C(CC(C)(C)C)(C(=O)N1CC=CC(NC(C2CCSC2)=O)C1)OC N1(C(c2n(C)c(S)nn2)=O)CC2CCN(C(c3ccc(F)cc3Cl)=O)CC12 N1(C(C2C(CC)N(C(C34CC3CNC4=O)=O)CC2)=O)CCC(F)C(O)C1 CC(C(=O)O)C(C)(O)C(=O)NCCC1CC(Cc2ccccc2F)C1 c1(C(=O)NCC2C(C(=O)Nc3cc(C)cc(F)c3)CCC2)cc2cccnn2c1 N1(C(C2(c3cc(C)no3)CC2)=O)CCCCC(NC(C2CSCCS2)=O)C1 C(=O)(C1=CC2(CCN(C(=O)C(C)C(C)COC)C2)C1)NCC1(C#C)CCCC1 CCC(C)CC(=O)C(=O)N1CCC1CC(N1CCCC(C)(C)C1)=O C#CC1CCN(C(C2COC(CNC(=O)C(O)C3CCCC3)C2)=O)C1 N1(C(CSC)=O)CC(C(F)(F)F)OCC1CNC(c1cc(C)c(CO)cn1)=O C(=O)(CCC(C)=O)NCC(COC)(F)F.C1(Cn2cc(C)nn2)OCCC1CSC C#Cc1cnn(CC(N2CCC(C(=O)NC(C)Cc3cccs3)(CF)C2)=O)c1 C(=O)(C(C)(C)C(C)(C)O)N(CC(C)(C)CNC(c1cn(CCO)nn1)=O)C c1(C(=O)NCCCC(C)(C)NC(C2C(=C)CC2)=O)c(C)ccc(Br)c1N c1(OCC)ccc(-c2cn(CCC(=O)NC3CC(O)C(F)C3)nn2)cc1Br c1(C(=O)NC(C2CCN(C(=O)Cc3sc(O)nc3O)C2)C)cncc(C2CC2)c1 c1(C(=O)NCC2CCC(NC(=O)C3=COCCO3)C2)cccc2ccsc12 c1(C(=O)OCC)cc(CNC(c2csc(Cl)c2)=O)ccn1.C1CC1CNC=O c1(C(N2CC(NC(C3(OC)CC3)=O)C2)=O)ccnc(C)c1Cl C1(CC)CCCN(C(=O)CC(C)(C)N(C)C(c2cc(C)c(C)[nH]2)=O)CC1 c1(C(N2C(C(=O)NC(C#C)C)CC3CC32)=O)cc(Br)c(C)c(Br)c1 NS(=O)(=O)c1ccc(CCCNC(C2CC2c2cc(F)ccc2F)=O)cc1 N1(CC(=O)Nc2scc(-c3ccc(CC)cc3)n2)CCC2(CC1)CC(C)NC2=O C(CCN(C)C(c1ccc(C)nc1O)=O)(C(C)(C)C)NC(CCC(=C)C)=O c1(C(N2CC(C)N(C(=O)C(c3ccc(O)cc3)=O)CC2)=O)cccc2nsnc12 c1(CNC(C2(COCC)CCC2)=O)n[nH]c2c1CN(C(=O)CCCC1CC1)CC2 Cc1nc(C)c(F)c(=NCC2C(C)CCCN2C(c2cn(C)ccc2=O)=O)[nH]1 C1(C(C(=O)NCC(C)N(C(=O)CCOCC=C)CC=C)F)CCOCC1 C1(CNC(CCCCCC)=O)(NC(=O)CC(C)CN(C)C)CCC(F)(F)CC1 C(CO)(CCCCNC(=O)C=C1CC1)NC(CCOC(C)C)=O CN1CC=CCC1CC(N1CCC=CC1C(=O)NC1CCCC(O)C1)=O CCC(O)C(C)C(=O)NC1CC2(C1)CC(C(=O)NC1CC(CCF)C1)C2 C1(CCC)(COC(=O)NCC2CCCN2CC)CC(=O)C1 Cc1cncc(C(=O)NCC2C(C)CCN2C(c2c(Cl)cnn2C(C)C)=O)n1 C#CC1(C(=O)NCCCN2CCC2)CCN(C(=O)CC2(COC)CC2)C1 C12(C(N3CC(N(C)CC4CCCN4Cc4ccccc4)C3)=O)CCC(CC1)CC2 N1(C(CSCCC(C)C)=O)CCCC1CN(C(C1CC1(Cl)Cl)=O)C1CC1 C1(NC(c2cc(C)no2)=O)(CO)CCCN(C(c2ccnnc2O)=O)C1 N1(C(CCCCC=C)=O)CCCC2(NC(c3cccn4nnnc34)=O)CC2C1 c1(C(N2CCC(C3CCC3)C2)=O)c(Cl)nsc1Cl.c1(CS)cncnc1-c1ccccc1 C(=O)(C1=NNC(=O)CC1)N(CCCNC(C1CC2(C)OCC1C2)=O)CCO Cc1ccc(C(N2CC(C(=O)N(C3CC4CC4C3)C)C2)=O)cc1F.CCO C(=O)(CC(C)(C)C(F)F)NC(C(C)C)CCN(C(=O)C(C1CCCCC1)F)C C#Cc1ccc(C)c(NC(C2CCC(C)CN2C(c2ccc(F)s2)=O)=O)c1 CC1CCN(C(c2cncs2)=O)C1CNC(c1cc(Br)n[nH]1)=O C1(OC)CC(CCNC(c2cc(C3CCC3)no2)=O)N(C(=O)C(C)CO)C1 N1(C(CC#C)=O)CCCCC1CNC(c1cncc(Br)c1)=O c1(NC2C(SC)COC2)ncc(S(=O)(=O)NCc2cccnc2Br)cc1Cl N1(C(C(C)CN(C)C)=O)CC2(CNC(c3ccc(-c4cccs4)o3)=O)CCC1C2 c1(C(=O)NC2CCN(C(c3ccn(C(C)C)n3)=O)C2)n[nH]c2c1CCOC2 C=CCC(CNC(c1cnc(S)nc1)=O)C(=O)N1CCC(O)(CC(C)C)C1 c1(C(C)C(=O)NC2CC2NC(=O)CC2=NNC(=O)C2)ccc2ccccc2c1 N1(C(Cc2n(C)ccn2)=O)CC(O)CC1C(=O)NC1CN(C(N)=O)C1 C1(NC(C(C)NC(CC)=O)=O)CC(NC(c2ccc(F)cc2)=O)C12CCC2 C1(CNC(C=CCC)=O)CC(NC(c2ccn(CC)n2)=O)C(O)C1 c1(OC)c(C(=O)N(C)CCNC(c2ccc(C)nn2)=O)cc(Cl)cc1C N1(C(CC2(OC)CC2)=O)CCCC2(C1)CN(C(=O)C(C)N=[N+]=[N-])C2 C=CCC(C(=O)NCC1CC1(C)C)NC(=O)COCCCC N1(C(c2occ(C)c2C)=O)CCC2CC1CN(C(c1cnn(CCF)c1)=O)C2 C12(C(=O)NC(CCNC(c3cc(C(C)C)nn3C)=O)(C)C)CSCC1C2(F)F c1(C(=O)NCC2COCCN(C(c3ncc[nH]c3=O)=O)C2)cncc2nc[nH]c12 c1(C(=O)NCC2CCN(C(c3cc(COC)on3)=O)C2)c(C)cc(O)cc1C Cn1cc(C(=O)NC2CCN(C(C3CC3Cl)=O)CC2)c(-c2ccoc2)n1 CCC(CCOC)C(=O)NC(C)CNC(c1c[nH]cc1-c1cc(F)cc(F)c1)=O C1(C(N2CC(OCCOC)C2)=O)CC1C1CN(C(=O)CCn2cccc2)C1 Cc1cccc(C(=O)NC2(CCNC(C3CC3C3CCCO3)=O)CCCC2)c1 c1(NC(=O)NC(c2ccc(C(=O)OCC)cc2)C)nn(C)c2c1CNCC2 C1(NC(c2c(C)nc(O)[nH]2)=O)COCCN(C(=O)C=CSc2nc[nH]n2)C1 N1(C(CC=C)=O)CCN(C(c2cc(=O)n(-c3ccc(C)cc3)[nH]2)=O)C2CCC12 CCC(CC)C(C)C(=O)N1CC2CC2(CNC(C2CC(n3ccnn3)C2)=O)C1 c1(C(=O)NCCOC2CCN(C(C(C3CC3)SC)=O)C2)cc(O)nc(O)n1 C12(CNC(C(CC)C)=O)CCCC1N(C(c1ccc(Br)c(F)c1)=O)CC2 C(=O)(C(CC(F)F)NC(c1nccnc1N)=O)NC(C#C)CC(C)C C(=O)(C(CC(=O)OC)NC=O)NCCC1CC(NC(CSCCCC)=O)C1 c1(OC)ccc(C(N2CC(CNC(C3CCN3C(C)(C)C)=O)C2)=O)cn1 CC(F)(F)C(C)(C)C(=O)NC1CC2CC(C1)N(C(=O)CCOc1ccccc1)C2 C=C(C)CN=c1cc(C)[nH]c(=NCc2cccc(S(C)(=O)=O)c2C)[nH]1 C(=O)(CCC1=CCCCC1)N(CCNC(C=C1CCC(C)C1)=O)CCOCCO C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCN(C(=O)CC2CCNC2=O)C1 CCS(=O)CC(=O)NC1CCN(C(c2cccc(C(C)(F)F)c2)=O)C1C(C)(C)C N1(C(C2(F)CN(Cc3ccncc3Cl)C2)=O)CCc2nc[nH]c2C1 c1(C(N2C(C)CC(CNC(c3cc4scnc4[nH]3)=O)C2)=O)ccc2nn[nH]c2c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2CCCN(C(=O)CN(C)C(C)=O)C2C1 c1(C(N2C(CC)CN(C(C3(CO)CCCCC3)=O)CC2)=O)ccc2n[nH]cc2c1 c1(SC)nc(N2CC3CC3(C(N3CCN(C(C)C#N)CC3)=O)C2)c(Br)c(C)n1 c1(C(N(C)CC2CCCN(C(c3cn(CC)nn3)=O)C2)=O)cnc2n1CCC2 C1(CNC(C(CC)O)=O)(NC(=O)CCCSCC)CCCCC1C.C(C)(=O)CC N1(C(c2c(C)nn[nH]2)=O)CCC(NC(=O)Cc2nc[nH]n2)C(CO)CC1 C1(C(N(C2CCN(C(CCc3c(C)nn(C)c3)=O)C2)C)=O)OCCN(C)C1=O c1(CNC(=O)Nc2c(C)nc(Br)cc2)cccn2ccnc12 C1(CC(N2CC(O)(C(C(N3CCC(N(C)C)C3)=O)F)C2)=O)CCCCN1C C(C(C)(C)C1=CCCC1)NC(C(CC1CCOCC1)NC(CSC(C)(C)C)=O)=O C(C)(CO)(C(=O)NCC(O)C(=O)NCC1CCC(F)(F)C1)OC c1(NC(C(=O)N(CC(n2ncc(C)c2)C)CC2CCOC2)=O)nc(Br)ccc1C CC1OCCC1(C)C(N1CC(NC(=O)COCc2ccnc(O)c2)C1)=O c1(N2C(CCCNC(c3cccc(F)c3F)=O)CCC2)ncnc2c1SCCC2 N#Cc1cn(CCC(=O)OCCCC2NC(=O)NC2=O)c(=O)nc1O N1(C(CCC2(C)CC2)=O)C2CCC1CC(NC(=O)CC13CCCC1C3)C2 C(=O)(CCC(C)Br)NCCCN(CC(=O)NCC#C)C Cc1cccc(C)c1OC(=O)CCCCCc1ccccc1.c12ccc(o1)CNC2 N#Cc1cc([N+](=O)[O-])ccc1NC(C1CN(S(=O)(=O)CCCCCl)CCO1)=O C12(NC(=O)CCSC(F)(F)F)CCCN(C(=O)Cc3cnoc3)CC1C2 CC1SCCC1(c1nnnn1C(C)(C)C)NC(c1cccs1)C1CCC1 CC1CC(O)CCN(N2CCC(C(N3CCOCC3)=O)CC2)C1 C1(C(=O)NCCN(C(CCSCC(C)C)=O)CC(C)O)CCCC(O)C1 N1(C(C(CC)OC2CCCC2)=O)CCC(C2CCCCN2C(C2OCCO2)=O)CC1 CC(=O)CCCC(C)C(=O)NCCNC(C1CCOC(C)C1)=O C1(C)(C(=O)NCC2(CNC(C3CC(C)OC3=O)=O)CC2)CCC(F)(F)CC1 Cc1cc(C(N2CC(O)CC2(C)C(F)(F)F)=O)ccc1S(=O)(=O)C(C)C C1(NC(CCCCC)=O)CCCCCN(C(c2ccn(C(C)(C)C)n2)=O)C1 C1(NC(CCSCCC)=O)CCN(C(c2ccccc2C)=O)C12CCC2 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCc2ccc(C)cc2)=O)CC1C c1(Oc2cc(CC(=O)N(C3CC4(CCC4)C3)C)[nH]n2)ccccc1C(F)F c1(NC2CC(CCNC(CC(CN(C)C)O)=O)C2)nc2c(cc1C#N)CCOC2 c1(CCC(N2CCC(NC(C(C(C)C)C)=O)(CO)C2)=O)ccc2ncccc2c1 N1(C(CC(C(=C)C)OCC)=O)Cc2occ(C(NC[Si](C)(C)C)=O)c2C1 CCC(C)C(O)C(=O)NCC1(c2ccccc2)CCN(C(C2CC2F)=O)CC1 N1(C(C(COCC)C)=O)CCC2(C=C(C(=O)N(c3cc(C)on3)C)C2)C1 CCC(CCOC)C(=O)N1CCC(C)(CNC(c2cc(Br)cnc2N)=O)C1 CC1(C)CCC(NC(C2COCCC2NC(=O)Cc2cncs2)=O)C1 c1(OC)ccc2cc(CNCCNc3cc(C)n(-c4ccc(Cl)cc4)n3)ccc2n1 C1(C(N2CCC(C)(NC(C(C)c3ccco3)=O)C2)=O)CCc2ncnn2C1 C1(CCOC)CN(C(=O)COC(F)(F)F)CCN1C(c1cc(Cl)c(Cl)s1)=O c1(C=O)cc(C#N)ccc1OC(F)F.Cc1ccc(N2CCN(C=O)CC2)c(C)c1 N1(C(c2ccc(=N)[nH]c2Cl)=O)CCC2(CC1)CN(C(C1CCCCC1F)=O)C2 c1(NC(c2nccc(OC)c2)c2nnnn2C(C)C)ccc(Cl)c(F)c1 c1(CN2CCN(C(C(C)NC(c3ccoc3)=O)=O)CC2)c(F)cccc1Cl C(=O)(C(C)(C)S(C)(=O)=O)NC(CN(C(C12CCC(CC1)O2)=O)CC)C Cc1ccc(SCC(N2CCC(CNC(c3occ4c3CCC4)=O)C2)=O)c(C)c1 c1(CC)cc(C(N2CCC(F)(CNC(C3CC(=O)N3)=O)C2)=O)nn1C c1(C(=O)NC2CC(C(=O)NC(CC)CC)CC2O)ccc(CO)c(F)c1 c1(CCC#N)ccccc1C(=O)NCC1(O)CC(CNC(=O)C#CC2CC2)C1 C1(NC(CO[Si](C)(C)C)=O)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 c1(OCC)cccc(CCC(=O)NCC2(O)CCN(C(=O)C=C(C)C)C2)c1 c1(CC(=O)NC2CCCN(S(=O)(=O)c3ccoc3)CC2)ccc(F)cc1Cl C1(NC2(c3n(C(C)C)nnn3)CC3CCC(C2)O3)CCCC2(CC1)CC2 CC1(C)OCCC1CC(=O)NCCCC(CO)NC(c1cccc(CO)c1)=O C=C(C)CC(C)C(=O)N1CCN(C(c2occc2COC)=O)C(C)C1 N1(C(C(C)OCCC(C)C)=O)CCCN(C(C2CC3CCC2O3)=O)CC1 N1(C(C=C2CCN(C)CC2)=O)CC2CCC1C1CN(C(=O)COCCCF)CC21 C(=O)(C(C#N)C(C)(C)C)NC1CC2(CC(NC(c3cc(CC)no3)=O)C2)C1 c1(C(=O)NC(C)(CNC(=O)CC2CSCCO2)Cn2cccn2)cccc(O)c1F C(=O)(CC(C)C(C)(C)C)NC(C(N1C(C)(CC)CC1)=O)Cc1cnc[nH]1 c1(SC)ccc(NC(=O)NC(C2(NCCC3CCC3)CCC2)=O)c(F)c1 N1(C(C(C)S(C)(=O)=O)=O)Cc2ccccc2C(CNC(=O)C2=NOCC2)C1 n1(CCC)cc(C(=O)NC2CC(F)(CNC(=O)C(O)CN3CCCC3)C2)cn1 Cc1nn(C(C)(C)C)cc1C(N1CCC(NC(=O)C=C(C2CC2)C2CC2)C1C)=O C(=O)(CCC(=O)NCC1CC(C)N(C(c2cc(COC)oc2C)=O)C1)NCC C(=O)(C1=C2CCCN=C2NN1)N(C)CC1CCN(C(C2CCCC(C)C2)=O)CC1 C(C)(C(C(=O)Nc1cnn(CC)c1)C(C)C)NC(CCC)=O c1(NC(C2c3ccc(o3)N2C)=O)ccccc1OC.C1(CC)CCC1C C1(N(C(=O)C(CC)N(C)C(c2cnc(Cl)s2)C)CC#C)CCN(C(C)=O)CC1 C12(NC(C)=O)CCN(C(c3ncc(Br)cn3)=O)CC1C2 CCCCC(CC(=O)N1CCC(C)CC1)NC(c1[nH]nnc1CC)=O C(CC(F)F)(C(=O)NCC1CC12CCCCC2)N(C(Cc1c(C)n[nH]c1)=O)C c1(NCCc2ccc(OC)c(C(C)(C)C)c2)ccc2ncn(C)c(=O)c2c1 C1(O)(CC(=O)NCCN(CCOCCCC)CCOC)CCCCC1 C1(CCC#C)CCCCN1C(=O)CN(C(=O)CN1CCCC(O)C1)C C1(Cn2cc(C3(N(C)C)CCCC3)nn2)COCCN1C(c1ccncc1O)=O c1(CC)nc(C)c(C(N2CCCCC2C(=O)NC(COC)CO)=O)o1 O=C(C1=CS(=O)CCC1)N1CC2(CCC(CNC(C3(CO)CCCO3)=O)O2)C1 C(CC(=O)N=c1ccn(C)[nH]1)c1cnc(N(C23CCCCC2C3)C(C)=O)s1 C(C(CC(=O)NCC1CC(NC(c2ccc3nn[nH]c3n2)=O)C1)C(F)F)N(C)C C1(C(N2C(C(=O)NC3(C(=O)OC)CCOCC3)CCC2C)=O)CC2C(C1)C2(F)F C1(C#N)(CSCC)CCC1.c1(C2C(=O)N2)ccnn1C.CC(C(F)F)=CC(=O)NCC1CC1 CC1C(NC(=O)CC2(C)CCCCC2)CCN1C(=O)C(F)CC1CCC1 C1(CNC(C(c2cccnc2)NC(CNC(N)=O)=O)=O)CC2(CCC2O)C1 N#CC1CCN(C(=O)COC2CCN(C(=O)CC3CCC(=O)N3)C2)C1 N1(C(C2CCC(=O)O2)=O)CC2CC(CNC(C3(C(F)(F)F)CCC3)=O)C2C1 NC(=O)C(F)(F)CNC(C1CC(NC(=O)COCC2CC2)C(O)C1)=O C(=O)(C(F)CCC(=O)O)NC(=O)C=CC(=O)N(C(C)C1CC1)C c1(CC)cc2c(CC(=O)NCC3(O)CCN(C(=O)Cc4cccs4)C3)csc2s1 C1(CNC(C(CC)NC(N)=O)=O)CC2CCC(C1)N2C(=O)CC(C)(C)OC C12(NC(CCCCCCC)=O)COCCC1CN(C(c1ccoc1C)=O)C2 N1(C(C2C(OCC)C2)=O)CCCN(C(=O)C2CC2)CC1 c1(CC)cnc(CNC2(C)CCCC2)o1.C1(NC(=O)N)CSC1(C)C c1(C(=O)NC(C2CCN(C(=O)CCc3cn[nH]c3)CC2)C)ccc(C2CC2)nc1 c1(C(=O)NCC2N(C(C3(CCOC)CCC3)=O)CC2)cn(C)c(=O)cc1C N1(C(Cn2ncc(C)c2)=O)CCC(C(=O)NC(c2cccc(O)c2)C)C(C)C1 C1(C(=O)OC)(NC(c2c(OC)n(C)nc2)=O)CCN(C(c2c(Cl)cnn2C)=O)CC1 C#CCCCC(C)C(=O)NCCCCCCN(C(=O)C=CC(C)(C)C)C C1(c2nnc(C)o2)CC2(CCN2CC2CC23CC3)C1 Cc1cnc(Cl)c(S(=O)(=O)N2CCCC(C)(C(=O)Nc3cnncc3Cl)C2)c1 c1(C(=O)NC(CC)CNC(=O)C(CO)N(C)C)n[nH]c2c1CCCC2 CCCCCS(=O)(=O)CC(=O)N1CCC(C(C)NC(c2csc(C(C)=O)n2)=O)C1 CCC(C)(C)CCCC(=O)N1CCC1CNC(=O)Cc1c(C)noc1C Cn1ncc(C(N2CCOCC2CC(=O)NCC2=CCCCC2)=O)c1Cl c1(C(C(=O)NC)N(C(CCCC)=O)CC)c(C)cnn1CC c1(C(=O)NC2(C#N)CCN(c3c(F)cnc(OC)n3)C2)c(Cl)cnc(Cl)c1Cl C(=O)(CCC(C)(C)C)NCC(c1ccc(C)cc1)NC(C(CC)C)=O CC1(C)CN(C(C2CC3CCC(C2)O3)=O)CCC1C(N1CC23CCC2(COC3)C1)=O CCC(C(=O)N1CCN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC1CF)C(C)(F)F C(=O)(CC(C)(C)C(F)F)N(CCOCCNC(c1cnc(SC)s1)=O)C CC(C)C(C)(CNC(=O)OC(C)(C)C)NC(c1ncc(Br)cn1)C S(=O)(=O)(c1cccnc1NC1CCCCC1C(C)(C)C)NCC(CN(C)C)(C)C c1(C(=O)NCC(C)(C)NC(c2n(CCOCC)ncc2)=O)nccnc1C(N)=O C(=O)(C(C(C)(C)O)NC(c1cnn2c1CCC2)=O)NCc1c(CC)nccn1 N1(C(C(C)(C)OC)=O)CCN(C(c2cccnc2-n2ccnn2)=O)C(C(F)F)C1 C=Cc1ccc(C(=O)N(CC(C)N(CCCCN(C)C2CC2)C)C)cc1 S(=O)(=O)(c1ccc(=NCC(O)c2ccnn2C)[nH]c1)N(CCN(C)C)CCO c1(C(=O)NCCNC(C2CC=CCC2)=O)ccnc2cc(F)cnc12 c1(C(=O)NCCC(CC2CC2)O)c(C(F)(F)F)cccc1F c1(C(C)C(=O)NC(C(=O)NCc2ccon2)C2CCC2)ccnn1C Cc1cn(C)nc1C(N1CC(C(O)C(N2CCC(N3CCC3)CC2)=O)C1)=O Cc1cc(NC(=O)CCc2cnn(C)c2)ccc1NC(=O)CC1CCC1C C1(CCC)CC(C(=O)NCC(C(F)(F)F)N2CCOCC2)CCO1 C1(C(N(CC(C)NC(C2(C)CC2)=O)C)=O)CCc2nnc(Br)n2C1 CC(CCC(C)(C)C)C(=O)N1CC2=C(C1)CN(C(=O)CN(C)CCO)C2 C(=O)(CCCCCCN=[N+]=[N-])NC1CCC(CNC(C(CCC)(C)C)=O)C1 N1(C(CNC(C(C)N(C(C)=O)CCO)=O)=O)CCN(C(=O)CSC(F)F)CC1 C1(C)(C(=O)NC2(C#C)CCOC2)CN(C(c2cc(F)ccc2F)=O)C(C)(C)C1 c1(C(C(=O)NCCNC(C2CC=CC2)=O)(F)F)cccc(Cl)c1 N1(C(C2(CNC(c3cccc(C)c3F)=O)CC2)=O)CCCCC(F)(F)C1 N1(C(CSCC=C)=O)CCCC(N(C(=O)CN2CCCCC2=O)CC)CC1 C(=O)(C1=CCC(C)CC1)N1CCN(C(CNC(=O)NC)=O)C(CC2CC2)C1 c1(C(=O)NC(C(C)NC(=O)CCn2cnnn2)C)cccc(OC(F)(F)F)c1 C1(CNC(C(CC)SC)=O)(NC(=O)C=Cc2cnn(C)c2)CCCCC1 C(=O)(N=c1[nH]n(-c2ccccc2)cc1C#N)c1cnn(CCOC)n1 c1(OC)c(Cl)nc[nH]c1=NCCC1CCCN(C(=O)CC2CC(SC)C2)C1 c1(C(=O)OC)cnccc1N1CC(C)(NC(=O)CSC2CCC(=O)NC2=O)C1 Cc1cccc(N)c1C(=O)NCC1(CCNC(c2cc(C(F)(F)F)on2)=O)CC1 C1(NC(c2c(C)cns2)=O)CCOC(C(=O)NCC[Si](C)(C)C)C1 c1(CC)cc(NC(C2(CNC(=O)CC(CC)C3CC3)CC23CCC3)=O)ccc1F C1(OC)CC(CCNC(c2c[nH]nc2C(C)C)=O)N(C(=O)C(F)C2CCCC2)C1 c1(C(=O)NCC2CC(NC(c3cc(OC)ncn3)=O)C2)cc(F)c(F)cc1F C(=O)(CS(=O)(=O)c1ccccc1C)N1C(CNC(CC2(NC(C)=O)CC2)=O)CC1 C1(C)(C(N2CCC(CNC(c3cc(CCOC)on3)=O)C2)=O)CCNC(=O)C1 CCCC(CC)N=c1cc(C)[nH]c(=NCc2cc(C)cs2)[nH]1 C1(C(N(CC(=O)NC(C)(C)C2(N(C)C)CC2)CC)=O)CCC(CO)CC1 CCCCC(C)NC(C1CCN1C(c1cncnc1)=O)=O c1(C(=O)NC23CC(CNC(C(C(C)C)(C)O)=O)(OC2)C3)sccc1S(N)(=O)=O C1(C(N)=O)CC2CCCC2N1C(c1n[nH]c2cccnc12)=O Cc1ccc(C(C)C(=O)NC2CC(CNC(c3c(Br)noc3C)=O)C2)cc1 c1(C(C2CCCN2C2CCCC2)NC(=O)NC(c2ccno2)C)nnnn1C1CC1 c1(OCCOC)cc(N2CCC(C)C2CNC(=O)Cc2cnoc2)ncn1 c1(C(=O)NC2C(C)CN(C(c3coc(Cl)c3)=O)C2)ccc(F)c(O)c1F CCC(C)CC(C)C(=O)N1CC(CC)(NC(=O)CN(c2ccc(Cl)cn2)C)C1 c1(CNc2cc(C)nnc2)cnn2cccc2c1 C(N=c1[nH]c(=NCc2n[nH]cc2Br)c2cccc(F)c2[nH]1)C1(C#N)CC1 CC1CN(C(=O)C(F)(F)C(O)C2CC2)CCC1CCNC(=O)CN(C1CCC1)C C#CCCCC(C)C(=O)NC(CC(C)(C)C)C(=O)Nc1c(C)noc1CC c1(NC(N2CCCCC2c2nccs2)=O)ccc(CC(F)(F)F)cc1 c1(CC(N2CC(CCn3cc(CC=C)nn3)C2)=O)cccnc1C CC1(C(=O)NCC2CCCC(CNC(=O)C(N)=O)C2)COC(=O)N1 N1(C(C2COCCN(C(C(C(C)C)C)=O)C2)=O)CC2CCCCC12C N1(C(CN(C(=O)OCC)C)=O)CC(NC(C2NC(=O)CC2C)=O)C2(CCCC2)C1 C1(C(N(CC(=O)NCC)C2CC2)=O)CCN(C(c2cc[nH]n2)=O)C1 C1(O)(CNC(C(CCNC(C(C)(C)CO)=O)O)=O)CC2CCC1O2 C=Cn1nccc1C(=O)NCC1CCCCN1C(c1cnn(CC(F)F)c1C)=O S(=O)(=O)(c1cccc(=NCC(F)(F)C2CC2)[nH]1)NCC1(COC)CCCOC1 C1(C(N2CC=CC(NC(CC(C)n3ccnc3)=O)C2)=O)CCCC(=O)CC1 C12(C(=O)NCC3CC3)CCCC1CCC2.C12(CC1)CNC(=O)C1(CC1)C2 C(=O)(CCN=C(NCC(C)(C)CCOC)NCc1cc2ccccc2o1)NC C(=O)(C1=NOC2COCC12)N1C(C)CC(NC(=O)C=Cc2ccnn2C)CC1 Cc1cc2n(n1)CCN(c1cc(N3CCOC(C)C3)nc(S(C)(=O)=O)n1)C2 N(C1c2ccccc2C2CC12)C(=O)CC1CC2(CCOCC2)CO1.C1(N)CCC1 N1(C(C(C)OC)=O)CCC2(CCN(C(c3cc(N)ccc3C(F)(F)F)=O)C2)C1 C1(CC(=O)NCC(C)(C2CCC2)NC(CCSC)=O)C(=O)ON=C1C CCCCCCCCCCC(C)NC(c1cc(Cl)c2c(c1)OCCO2)=O C1(NC(c2c(C)ccs2)=O)CC12CCN(C(c1c(F)ccc(C)c1F)=O)CC2 n1(CC(=O)OC)c(C)cc(C(=O)NC(CNC(=O)CC23CCC(CC2)C3)CO)c1C C=CC(C)CCN=c1[nH]c2c(c(=NCc3cc(O)no3)[nH]1)CCCC2 C1(NC(C(C)CC2CC2)=O)(CO)CCN(C(c2conc2C(C)(C)C)=O)CC1 c1(C(CC)C(=O)N2CC(NC(c3ccc(CSC)o3)=O)C2)ccc(F)cc1 C1(C(N2CCC(C)(CNC(c3c(CC)nn(C)c3)=O)C2)=O)CC12CCN(C)C2 N1(S(=O)(=O)C2CC2c2cccc(Br)c2)CCn2ncc(C3=COCC3)c2C1 c1(C(N2CCCC(NC(c3cc(O)cc(O)n3)=O)CC2)=O)ccc2sccc2c1 N1(C(C)=O)CCN(C)C(CO)C1.c12cc(nn1C)C(=O)NC1CCN(CC1)C2=O N1(C(C(C)Cc2ccnn2C)=O)CCN(C(=O)CSc2cn[nH]c2)CC(C)(F)C1 N1(C(c2cccc(Cl)c2)C(=O)NC2COC2)CC(O)C2(CCCC2)C1 C(=O)(C1=NOC2(CCCN(S(=O)(=O)C(Cl)(Cl)Cl)C2)C1)NCCCCS(C)(=O)=O c1(NC(C2CCCC(C)C2)=O)ccc(Cl)c(C#N)n1.C12CCCN(C1)C2=O c1(C(C)(C)OC)cc(=NC(=O)CC(=O)N2CCC3(CC(O)c4ccccc43)C2)[nH]o1 CC1CN(C(C2C(C)(C)C2(C)C)=O)CC(C)C1NC(c1cc(Cl)c(Cl)s1)=O C1(C(CC)C)CCCN1C(=O)C(C)N(C(=O)CCN(C(N)=O)CCO)C N1(C(C2CCC(COCC)C2)=O)CC(C)(C)OCC1NC(=O)C(C)(C)C1CCC1 c1(C(=O)NCCC(C)CCNC(=O)CCCc2cnn[nH]2)cnn2c1CCCC2 C(C(=O)N1CCC(O)(CNC(c2ccc3c(c2)CC3)=O)C1)(C(C)(C)C)SC C1(COCC)CC(N2CCCCC2NS(=O)(=O)c2ccccc2)CCO1 N1(C(C#CC(=O)N(C)C)=O)CC(C2(NC(C3CCCNC3=O)=O)CC2)C1 c1(C(=O)NCC(C2CCCCC2)Nc2cc(CC)ncn2)cc2n(n1)CCCC2 N1(C(CCCC=C)=O)CC2CN(C(c3ccc(O)c(C)c3)=O)C2C1.N c1(C(=O)Nc2c(C)nc(F)cc2)n[nH]c2c1CN(C(c1sccc1CO)=O)C2 N1(C(CC(C)c2cccnc2)=O)CC2CC(C1)CN(C(C1CCCNC1=O)=O)C2 CCCCCC(C)(CC)C(=O)NCCCCCCn1cc(C2CCCC2)nn1 N1(C(CC(CC)CC)=O)CC2(CCC2)CC1CNC(c1c(C)ccc(C)c1C)=O C(C(C(F)(F)F)NC(=O)Nc1ccc(-c2cccs2)cc1)OC C1(CC(=O)NC(C(=O)OCC)C)CC2(C1)CN(C(=O)CN(C)C(N)=O)C2 CCCCC(CN=c1nc(O)c(Br)c[nH]1)NC(c1ccc(Cl)cc1C)=O C(=O)(N=c1cnn(C)[nH]1)C1N(C(c2cccc(OCC(=O)OC)c2)=O)CC(C)C1 C=C=CCCC(=O)NCCC(=C)CNC(c1occc1Br)=O c1(CN(C)C(c2ccc(O)cn2)=O)ccccc1CNC(c1cn(CCO)nn1)=O C1(NC(c2ccc(OC)o2)=O)COC2(CNC(=O)C(C)(C)CNC(C)=O)CC1C2 C=CCCCCC(=O)NC1(CC(=O)NCC(=O)N(C)C)CC1(C)C C=C(C)CC(C(=O)NC(C)CCC(=O)NCCc1ncoc1C)OC Cc1ccc2c(c1)CC(C(=O)OCC1CCCN1)S2(=O)=O CC1=C(C)CC(C(=O)NC2CN(C(C34CSC(C3)C4)=O)CC2C)CC1 CC1(NCCNC2(c3nnnn3CC(F)F)CCC2)CC(F)(F)C1 c1(COC(CNC)=O)nc(C)c(NC(c2ccccc2C)=O)s1 c1(C(=O)NCC(C(C)(C)C)NC(C2(NC(N)=O)CC2)=O)cc2c(nc1O)CCC2 N1(C(C2CN(C(N)=O)C2)=O)CC(C2CC2)(C(N2CCC(O)(C(F)F)C2)=O)C1 N1(C(c2[nH]c3cc(C(C)=O)sc3c2)=O)CCOC2CN(C(=O)C=CC(C)C)CC12 c1(-c2cnc(NC(c3cccc(OC)c3O)=O)c(O)c2)cccc2c1OCC2 C(=O)(C(O)C(F)(F)F)NCC=CCC(N1C(C(=O)NCC)CCC1)=O c1(C(=O)NCC2C3CN(C(c4nscc4Br)=O)CC23)cncc2sccc12 N1(C(CCC(=O)NCC)=O)CCCC(C(=O)NC(C)(C)C(=O)OC)C1C N1(C(CC(=C)Br)=O)CCN(C(c2nnccc2C)=O)C(C)C1C C1(NC(c2c(C)nsc2C)=O)CC2CC(C1)N(C(C1CN(C3CCCCC3)C1)=O)C2 S(=O)(=O)(c1cc(C(=O)O)cs1)NCC(=O)Nc1c(C)noc1-c1ccccc1 c1(C(C(=O)NC(C(=O)OC)C)N(C)CC2CC(=O)N(CC)C2)nc(Br)c(C)cc1F C1(CC(=O)NCC2(NC(CCc3cc(C)[nH]n3)=O)CCCC2)CCCCC1(C)C c1(C(N2CCCC2Cc2cn(C3CC3)nn2)=O)cccc(C(F)F)n1 C1(C(=O)NC(C2CCCN2C(=O)Cc2ccsc2)(C)C)CN2CCCN1CC2 C(N=c1[nH]c(N2CC3CC2C(F)(F)C3)nc2cccnc12)C1COC(=O)C1(F)F Cc1ccc(C(N2CC(NC(C3CCC(=O)NC3)=O)C(F)(F)C2)=O)cc1O c1(NC(CC(CCC)NC(=O)OC(C)(C)C)=O)ccc2ccn(C)c2c1 CC1(C)CC(NC(=O)CC(CNC(=O)Cc2cncs2)C2CCC2)C12CC2 Cc1cc(C(=O)NCC(C)(C)OCCNC(c2c(C)nc(C)n2O)=O)cc(F)c1 c1(CCC(=O)OC)ccc(CNc2ccc(C3(C)CC3(F)F)cc2)cc1 C(=O)(CCC(C)(C)C(=O)OC)N1CCC(OC(CNC(COCC)=O)C)CC1 N1(C(CC(CC)(F)F)=O)CCN(C(C2(C)CC(C)=NO2)=O)CC(C)C1 N1(Cc2c(C)nn[nH]2)CCC(C2CCCN(C(=O)C(C)NC(c3ccoc3)=O)C2)C1 C(=O)(C1=C(C2CC2)N(C)C(=O)N(C)C1c1cnc2c(F)cccc2c1)OC Cn1cnc2c1C(C(=O)N=c1ccn(Cc3ccc(F)cc3F)[nH]1)CCC2 C1(C)(CC)CC(NC(=O)CNC=O)CN1C(c1oc(C)nc1C)=O c1(C(=O)NC2C(NC(CC=C=C)=O)CC2)ccc(C#N)c(Cl)c1 c1(C(=O)NC(C(C)NC(=O)CC2CCCC2)C)ccc2c(c1)NC(=O)CCN2C C1(c2nnnn2CC2CCOCC2)(NC(CC(C)(C)C)C)CCC=CCC1 c1(-c2ccc(CC)cn2)nc2ccc(C(=O)Nc3ccc(C#N)cc3Cl)cc2s1 CCCC(CCC)CC(=O)NC(C)C(=O)Nc1ccc(CCO)cc1 CCCCCCCC(=O)NC1CC(C(=O)N(CC(=O)OC)C)=CC1O c1(C(=O)NC2CCC(C(=O)NCC3CCN(CC)CC3)C2)cc(F)cc(Br)c1F C1(C(=O)NC(CC)COC)CC2CCCC2N1C(C1CC(=O)N(C)C1)=O C1(NC(c2c(CC)nccc2)=O)CCCN(C)CC1 C(=O)(C(CNC(c1ncncc1Cl)=O)CC(C)C)NC(CC)CCOC C12(CNC(C3C(C=C)C3)=O)CCC(NC(=O)C(=O)NCC3CC3)(CC1)CO2 c1(CCOC(C)C(=O)NC2CN(C(=O)C(c3ccccc3)F)C2)ccccc1 c1(C(N(C(C(C)C)C)CCC#N)=O)cn(CCNC(=O)C(F)C2CCCC2)cn1 c1(OC)ccc(C(N2CC(CNC(=O)CCc3cnc(C)s3)C2)=O)cc1C1CC1 N1(CC(=O)NC2(C3CN(C(=O)CC=C(Cl)Cl)C3)CC2)CCCCC(O)C1=O c1(C(N(CCOC)CCNC(=O)Cn2cccn2)=O)c(F)cc(C)cc1F C12(C(=O)NC(C)C(C)n3cccn3)COC(C1)C(NC(c1cnc(CO)o1)=O)C2 c1(OC)oc(C)nc1C(N1CC(CNC(c2ncc(C(F)F)s2)=O)CC1C)=O CC1(C)CCN(C(=O)C(C2CC2)C2CC2)C1CC(=O)NCC(CO)C1CC1 C1(C(N2CC(c3ccccc3)(Nc3ncc(C(N)=O)s3)C2)=O)CC2(C1)CC(O)C2 C(=O)(C(CO)C(F)(F)F)N1CC2C(C(=O)NCCc3nc(C)[nH]n3)C2C1 C(=O)(C(O)CSC)N(CC(=O)N(CC(C)OC)C)CC1CC1 c1(C(=O)NCC2C(NC(c3cccc(C(C)C)c3F)=O)C2)ccc2c(c1)NCC2 C(=O)(CC(C(=O)N(CC(O)CNC(=O)CN1C(=O)CCC1=O)C)NC(C)=O)OC c1(C(N(C(C)CCNC(c2cc(Cl)cnn2)=O)C)=O)ccnn(C)c1=O c1(C(=O)NC2C(CNC(Cc3cn(C)nc3)=O)CCC2)cc2n(n1)CCCC2=O C1(C(=O)NCC(C)Cn2ccnc2)CN(C(C2(C(N)=O)CCC2)=O)CCO1 C1(C(=O)OC)CCCN(S(=O)(=O)N2CC(OC(C)C)C2)C1 CCS(=O)CC(=O)N1CCC(C)(CCNC(=O)Cc2ccnn2C2CCCC2)C1 c1(C(N(CCC(C)NC(c2c(SC)cnn2C)=O)C)=O)cc(N)cc(C)c1F N1(C(c2cn(CC)nc2)=O)CCC2CCN(C(=O)CC3=CCCC3)C2C1 C1(NC(C2C(C)CCO2)=O)CCCC(CC(=O)NCCc2cccn2C)C1 c1(-c2nc(O)cc(C)c2Br)nc(C2COc3ccccc32)nn1Cc1cccs1 Cc1nc(O)ccc1C(=O)NC1COCCN(C(C2CC2C)=O)C1 n1(CC(C)C)[nH]c(CC(=O)NCCCC(C)NC(C2CCCOC2)=O)cc1=O C1(C(N2CCC(O)(CN(C)C(C3CC4(CCC4)C3)=O)C2)=O)CN2CCN1CC2 C#CCCCCC(=O)N(CCNC(C1CC1c1ccc(F)cc1C)=O)CCOC S(=O)(=O)(CC(=O)NCCCN(C(=O)C(=O)Cc1ccccc1)CCO)N(C)C N1(C(C2C(CC)CCC2)=O)CC2CC(C1)CN(C(c1cnc(S)nc1)=O)C2 C(=O)(C1CCCc2ccnn21)N(C1CCCN(C(c2c[nH]c(=N)s2)=O)C1)CCO CCC(C)(CNC(c1n[nH]cc1Cl)=O)NC(C1CC(=O)C1C(C)(C)C)=O c1(N(C)C)cnc(C(N2CCCC(CNC(c3cocc3C(N)=O)=O)C2)=O)cn1 c1(OC)cc(Cl)c(Br)cc1NC(CCC(C)C)C(=O)OCc1nnnn1C C1(C(=O)NCCC2(CNC(C(C)OCC=C)=O)CC2)CCOCC=C1 N1(C(C2C(C)OC(C)C2)=O)CC2(CCCC2NC(c2noc3c2COCC3)=O)C1 Cc1c(C(N2CC(CNC(C3(C)CC(C)OC(C)C3)=O)C2)=O)cccc1[N+](=O)[O-] N1(C(c2c(C)nns2)=O)CC2(C)CC1C2NC(=O)C(C)Cn1cccn1 N1(C(C2CCN(CC)C2)=O)CCC(NC(c2snnc2C2CC2)=O)C12CC2 C(=O)(C(C)S(N)(=O)=O)N1CC(C(=O)NC(c2ccncc2)C)C(C)C1 c1(N(CC(=O)OC)C)ncc[nH]c1=NCc1ccc(-c2cccc(CO)c2)cn1 c1(C(C)C)ccc(C(=O)NC(C)CC(C)NC(c2ccc(COC)cc2)=O)cc1 N#CC1(C(=O)C(=O)NC2CC2CNC(C2(N3CCCC3)CC2)=O)CCC1 n1(CCC(N2CC(OC)(CNC(=O)CCC3(C)CC3)C2)=O)cnccc1=O C1(CN(C(c2coc(C(C)(C)C)n2)=O)CC)CCCCN1C(=O)C1=COCC1 c1(C(N(CCCCN(C(=O)CCc2cnc(O)[nH]2)C)C)=O)cccc2nsnc12 c1(CN(CC(=O)OCCn2cccn2)C)cc2c(cc1O)OCCO2 c1(CNc2c(CC(N3CCC(F)CC3)=O)cccc2)cccc2nccnc12 C1(C)(C(N2C3(CNC(CCC4(C)CC4)=O)CC(C2)C3)=O)CC(C(F)(F)F)=NO1 C(=O)(C(C(C)(C)C)N(C)C)N1C(C(N2C(C=C)CC2)=O)CSCC1 c1(C(N2CC(NC(C3(C=C)CC3)=O)C(OC)C2)=O)ccc(C(F)(F)F)cc1CC CCC(CNC(=O)CC1OCCC1C)(CC)NC(c1cnn(CC2CC2)c1)=O C1(CNC(c2ccc(COC)nc2)=O)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 C1(N(C(Cc2scc(C)n2)=O)C)CCCN(C(C2CNC(=O)N2C)=O)CC1 N1(CC=C)CCC(C(=O)OC(C)CS(=O)(=O)CC)c2ccccc21 C1(NC(C(C)NC(=O)NC)=O)CCC2(CCN(C(=O)CSc3cn[nH]c3)C2)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)N1CCC(C2(NC(C(COCC)C)=O)CC2)C1 N1(C(C2N(C(C)=O)CC(O)C2)=O)C2CCC1CC(NC(c1ncccc1Cl)=O)C2 C1(CNC(C2(SC)CCC2)=O)CCC2(CN(C(=O)C(=CC3CCCC3)C)C2)O1 C1(CNC(CC2(CNC(C(F)=CCC)=O)CC2)=O)OCCC1(C)C Cc1sc(-c2ccc(OCC#N)cc2)nc1NC(N1CCOCC1CC(C)C)=O Cc1cc(C(=O)NCC2COCC2NC(=O)CCC2=NNC(=O)C2)c(C)c(C)c1 N1(C(COCP(C)(C)=O)=O)CCC(C2CCN(C(c3coc(Cl)n3)=O)CC2)C1 C1(C#CC(=O)N2CCC(C(C)NC(c3nc(C)ccc3C)=O)CC2)(CC)COC1 Cc1cccc(CCC(=O)NC2CCC(N(C)C(C3NC(=O)OC3C)=O)CC2)c1 C(CC(C)C)(C(=O)OC)NC(C1(C(c2nnnn2C2CCOC2)SC)CCC1)(C)C C12(NC(Cn3c(C)ccn3)=O)CC(C1)N(C(c1cn(C3CCOC3)cn1)=O)C2 c1(C(N(C2CN(C(C(C)=C(CC)C)=O)CC2F)C)=O)cc(F)c(F)cc1OC c1(C(=O)NC(C)(CO)C(=O)N2CCC(n3ccnc3)C2)cccc2cc[nH]c12 C1(CCC)CN(C(c2cn(C)nc2OC)=O)CCN1C(=O)CC1CCC(=O)N1C c1(OC)cccc(CNC(c2c[nH]nc2CCNC(=O)C(C)OC)=O)n1 c1(CC(C(=O)NCC(CNC(C2CC(CC)C2)=O)O)O)cccc(OC)c1 c1(C(N2CC(CNC(c3n[nH]c(C)c3F)=O)C(O)C2)=O)cc(Cl)c(F)cc1F c1(C(N2CCC(C(=O)NC(COC)C(C)C)C2)=O)c(OC)cccc1C Cc1cc(F)ncc1CNC(=O)CCN(C)C(C1CCN(C)C(=O)C1)=O S(=O)(=O)(c1cccc(-c2ccnn2C)c1)NC(c1noc(CN)n1)C CCC(CC)CCC(=O)NCC1CCC1NC(c1cccc(C(F)F)c1F)=O N1(C(C2(C)CC=C(C)CC2)=O)C2CCC1CN(C(c1nnn(C(C)C)c1C)=O)C2 c1(C(=O)NCCC2OCCCN(C(C(C=C)O)=O)C2)cc2ccccc2c(=O)o1 CCS(=O)c1ccccc1C(=O)NCCC(F)(F)Cn1cc(C2CC2C)nn1 C1(NC(c2ccc(CCC)s2)=O)CC2CCC1C(NC(=O)C#CC(C)(C)C)C2 C1(C(CC)C)CCN(C(=O)C(F)C2CC(NC(C3CC3C#N)=O)C2)CC1 N1(C(CC2C(CC)C2)=O)CC(NC(C2(C)CCCN(C)C2)=O)C(N=[N+]=[N-])C1 c1(NCCC(CC)C)[nH]c(=NCc2ccc(NC)cn2)nc2ncn(CC)c12 C1(CC)CN(C(=O)CCCN(C(=O)COC2(C)CCC2)C(C)C)CC(CC)O1 C1(NC(c2c(CC)cccc2)=O)CN(C(=O)C(O)C2CCC2)CC1S(C)(=O)=O c1(C(=O)NC23CC(CNC(c4n(C)ncc4)=O)(C2)C3)nccc(F)c1Cl N1(CCN(C(c2c(CSC)c[nH]n2)=O)C)CCN(C(=O)C(C(C)O)N(C)C)CC1 c1(C(N2C(C(N(CC(CC)CC)CC)=O)CC2C)=O)cc(C)nc(C)n1 N1(CC(=O)Nc2ccccc2C(F)(F)F)CCN(C(=O)C=CCBr)C(CCO)C1 CC1=C(c2ccc(CCC(=O)NCC3(C)COC3)cn2)CCCC1 c1(NC(COc2cccc(OC)c2)=O)ncnc(C(F)F)c1Br C1(C(NNC(=O)C2CCN(C(C)=O)C2)=O)CCc2ccccc2O1 N1(C(CCCCCC)=O)C2CCCC1CC(CNC(=O)Cc1cncc(F)c1)C2 C1(OCC)CC2(C1)CC2NC(C12CC1CN(C(c1cnc(N(C)C)o1)=O)C2)=O Cc1cc(C(=O)NCC2CCN2C(=O)C(O)CC#N)n(SC(C)(C)C)n1 c1(N(CC(=O)N(CC(O)CNC(c2c[nH]c(=O)cn2)=O)C)C)ccc(Cl)cn1 c1(C(N2CCC(O)(C(C)NC(CNC(C)=O)=O)C2)=O)c(C)ncc2ccccc12 c1(N(CC(F)(F)Cl)C)nc(N2CCN3CC4(CC4)CC3C2)nc2ccsc12 CC1=NN(C)C(=O)C1CC(=O)NC1(CNC(c2cn(C)cc2C(F)(F)F)=O)CC1 c1(C(=O)NCC2CCC(NC(c3cc(CC)no3)=O)CC2)cnn2cnnc2c1 C(c1ccncc1)=C(C(=O)NCC(CC)NC(=O)C(C)CN1CCOCC1)C N1(C(c2cc(C)ncn2)=O)CCOCC(NC(=O)CC(O)C(C)C)C1 C1(C(=O)NCC2(C(=O)NCCOC3(C)CCC3)CCCC2)CC12CCOCC2 Cc1cc(Cl)c(Cl)cc1C(N1CCOC(CN(C(=O)C=CCN(C)C)C)C1)=O N1(C(CC2CN(C(C(C3CN(C(C)=O)C3)OC)=O)C2)CCC)CC(F)(F)CC1C C1(NC(C2(C)CCCN(C(=O)CN3CCOCC3=O)C2)=O)CCCOC12CCC2 c1(C(C)C(N2C(CNC(=O)C3=COCCO3)CC(O)C2)=O)c[nH]c2ccccc12 C=CCC(CC(C)C)C(=O)NC1(C(=O)NC2CC2O)CCC1 C12=CC=C(C=C1)C2.CC1CCC(C(=O)N(CCNC(c2n[nH]cc2Cl)=O)C2CC2)C1 C1(NC(c2c(COC)scc2)=O)CN(C(c2n[nH]cc2C)=O)C2(CCOC2)C1 c1(C(N2C(C)(CNC(Cc3ncc(C)o3)=O)CCC2)=O)ncnc2c1CCCC2 CN1CC2(CCN(Cc3ccc(F)c(-c4ccc(F)cc4CO)n3)CC2)C1 C1(NC(c2nccc(C)c2)=O)CN(C(=O)C2=CS(=O)CCC2)CC12CCC2 N1(C(c2c(OC)ccs2)=O)CCC(C)C(NC(=O)COc2cc(F)cc(F)c2)C1 c1(CC)cnc(Cl)[nH]c1=NCC1CN(C(c2c[nH]nc2C(C)C)=O)CCO1 C1(C(=O)NC(CNC(C(c2nc(C)sc2)=O)=O)C(C)C)CC2CCC1O2 Cn1nc(C(=O)NCC2CN(C(c3ccc(C(N)=O)cc3)=O)CC2O)ccc1=O CC(CCC(=O)N1CCC(O)(Cc2cnns2)C1)N(C)C.C1C(=O)N1 c1(OC)ncnc(C(=O)NCCCC(C)(C)NC(=O)CCOCC2CC2)c1F C#CCCCC(C)C(=O)N1CCC(C2CC2)(NC(=O)Cn2cnnc2O)C1 N1(C(C(=O)NCC)=O)CCn2c(CNC(C3CC(=O)C3)=O)nnc2C1 N1(C(c2nn(C)cc2I)C(=O)NCCCOC)CCCCCC1c1ccncc1 N1(C(c2nc(C)n(C)n2)=O)CC2CC(NC(c3ccc(N=[N+]=[N-])cc3)=O)CC1C2 C(=O)(C1=CCCSC1)NCCC(C(=O)N1CC(COC)C1)O C1(NC(c2cncc(OC)c2)=O)CC2CC(NC(c3cc(C)n(C)n3)=O)CC2C1 c1(C(=O)NC2C(NC(c3c(=N)cc[nH]c3)=O)CCC2)coc2cc(F)ccc12 CCCCCCC(C)CC(=O)NC1C2CC1N(C(=O)CCn1nc(C)nc1C)C2 C1(CN(C(=O)CC2(C)CC2)C)CCCCN1C(=O)Cc1ccccc1Br O=CCCCn1cc(CNC(C2CCCC2)CO)nn1.N1(C)CC2CC2C1 C1(C2CCCCC2)(NC(C(C2CCOC2)NC(C2C(OC)(OC)CC2)=O)=O)CC1 CC1CCC(F)(C(N2CCCC2CCNC(=O)Cc2cccc(F)c2)=O)CC1 C(=O)(C1CCc2nccn21)N(C1(C(=O)NC2CCCCC2)CC1)C C=C(Cl)C(C)(C)C(=O)N1CCCC(N(C(=O)Cc2cccc(Cl)c2F)CC)C1 CN=c1nc(N(C)CC2CCN(C)C2)[nH]c(=NCc2cc(C)ccc2F)[nH]1 CCC(CN=c1cc[nH]cc1S(=O)(=O)NCCS(=O)(=O)CCO)c1ccccc1 c1(CCC(=O)NCC(CO)NC(C2(C(C)C)CCC2)=O)c[nH]c(=N)[nH]1 Cc1ncccc1C(=O)NC(C)(C)CN(C(=O)Cn1cccnc1=O)C c1(C(N2CCN(C(C(CC#C)C)=O)CC2CCC)=O)cc(F)cc(C)c1O CC1(NC(=O)Cn2cc[n+](C)c2)CCCN(C(=O)CCCc2cccc(Cl)n2)C1 Nc1ccc(CCC(=O)NCCCCCCNC(=O)CN2CC3CC3C2)nc1 O(NC(=O)C(C)(C)C(C)NC(=O)C(C)c1ccco1)CCOC C12(NC(c3c(C)n(C)nc3)=O)CCC(CNC(c3nccc(Cl)c3F)=O)(C1)OC2 N1(C(c2c(C)nn(C)c2N)=O)CCC2(CC1)CN(C(c1occc1Cl)=O)C2 N1(C(=O)CC2CNC(=O)O2)CC2CC(C1)N2C(C1(O)CCCC1)=O c1(C(=O)NCC(C2CC2)NC(C(C)OCCOCC)=O)ccc(N)c(Cl)c1 CC1N(C(=O)CNC(=O)CC2COC(=O)C2)CCCC1(C)C N1(S(C)(=O)=O)CC2CCC1CN2C(c1cnc(Cl)c2c1OCO2)=O C1(CCC)CCCC1NC(c1cc(CNC(=O)CN(C)C(=O)C2CC2)cs1)=O C1(COC(c2ccc(SCC)nc2)=O)CCN(c2ncnc(OC)n2)CC1C C=C1CCC(C(=O)N(C2CCCN(C(=O)C(F)OC)C2)CCF)CC1 C12(C(=O)NCC(CCOC)NC(c3nnc(C)s3)=O)CCC(CC1)CC2 C1(NC(C2(COC)CC2)=O)CC2(CCCCN2C(C2SC3C=CC2CC3)=O)C1 N1(C(C(C(C)C)NC(C)=O)=O)CC2(CC(NC(C3CC(F)(CO)C3)=O)C2)C1 C1(C(=O)NCCN(C(C2C(OCC)C2)=O)C2CC2)CCC(O)CC1 c1(CC)cc(NC(=O)C(=O)N(Cc2cn(C)nn2)C)on1.C1(C(=O)N)CCCO1 c1(CCC(=O)NC2C(NC(CCC#CC)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2c(SC)scc2)=O)CCC2(CC1)CN(C(=O)C(C)CCCC(C)C)C2 N1(C(=O)NC2CCC(C)CC2)CCC(C=CC(=O)NCC(C)(F)C(C)(C)F)CC1 N1(C(C(=O)Nc2ccc(OC)cc2)=O)CCC(C)C(NC(C2COC(C)C2)=O)C1 C(C(=O)NC(=O)C(C)(F)F)(C(C)C)NCC1(CC(=O)OC)CCCCC1 C1(NC(c2cnc(C)n2C)=O)CN(C(C2Cc3nccn3C2)=O)C2CCCC12 c1(C2C(C(=O)NCC3CCN(C(c4c(N)non4)=O)C3)C2)cccc(F)c1F N1(C(=O)CC2CCN(C(=O)Cn3ccnc3)O2)CC23CCC2(COC3)C1.O=C C=CCC(C)C(=O)N(CCNC(c1ccc(C(C)C)cc1)=O)CC1CC1 C(N=c1[nH]c(N2CCC(C)(CO)C2)nc2ccccc12)C1CCC(C)(C)CO1 Cc1nc(C)c(CC(=O)NC(C)CN(C)C(c2cc(N)ccc2O)=O)c(O)n1 N1(C(C(CCC)NC(c2ncn(C)n2)=O)=O)CCC(C)=C(F)C1 c1(C(=O)NCC2(CNC(c3cc(C(N)=O)on3)=O)CCOC2)ncncc1Cl N1(C(CCN2CC(=O)NCC2)=O)CCC(NC(C2CC3CCC2CC3)=O)C(O)C1 c1(C(=O)NC2CCCC(Nc3ncc(I)cn3)C2)cc2ccccc2oc1=O c1(C(=O)NCC2C(NC(c3n(C(C)C)ccc3)=O)CC2)cnn2cccnc12 N1(C(C(C=C)CC)=O)CCC(n2cccn2)(C(=O)NCc2ccc(=N)[nH]n2)CC1 c1(C(C(C)N(C=O)Cc2c(CC)cco2)O)ccc(F)cc1 Cc1ccc(C(N2CC(C(C)NC(c3c(C)coc3C(C)C)=O)C2)=O)c(C)c1 CC1CCCCN(C(=O)C(C(C)(C)O)NC(=O)C(C)C#N)C1 C1(CNC(C(C)NC(C2CCCC2)=O)=O)CN(C(=O)CC2CC2C)CCC1(C)C C#CCCC(O)C(=O)NCC1(F)CCC(NC(=O)CCCn2ccnn2)C1 C(=O)(C(C)(C)CC(F)F)NCCC(CNC(CCCCCOCC)=O)O CCCC(CCCNC(c1ccc(OC)cc1Cl)=O)NC(C1(Cl)CC12CCC2)=O N1(C(CSCCOC)=O)CCC(C(F)F)(CNC(=O)C(C(C)C)n2cncn2)C1 C1(C(=O)NCc2n(CCC)ccn2)CN(C)CCN1C(=O)CC1(N(C)C)CCC1 c1(C(N2CCC(CN(C)C(c3scnc3C3CCCC3)=O)C2)=O)ccccc1Cl C1(CSC)CCN(C(=NCc2sccc2S(C)(=O)=O)NC2CCS(=O)(=O)C2)C1 N1(C(CC(C)C2CCCC2)=O)CC2CCCCC2(NC(=O)Cn2ncnn2)C1 c1(-c2cn(CCC(C)NC(=O)CCN3CCC3)nn2)ccc(-c2ccco2)cn1 CC(C)(C)CC(C)(C)C(=O)NCC1CCC(NC(=O)COCc2nc[nH]n2)CC1 Cc1cc(C)n(CC(N2CCNCCC2c2ccccc2)=O)c(=O)n1 CCCC(O)C(CO)NC(=O)CN(C(c1cc(C)nnc1C)=O)CC1CC1 N1(CC(C)(C)NC(=O)C=Cc2cccnc2)CCN(C(C2CCNC2=O)=O)CC1 C1(NC(C2(CC=C)CCOCC2)=O)CCN(C(C2(C#N)CC2)=O)CC1F c1(N2CC(C)CC(CC)C2)ccncc1S(=O)(=O)N1CCCC(C(N)=O)C1 c1(OC)cc(C(=O)NC2CC2NC(c2c(Cl)ccnc2C)=O)cc(Br)c1 O=C(CCCCCc1cccs1)NCC1CN(C(=O)CC(O)C2CC2)CCO1 n1(CC)c(-c2nc(C3CCOCC3)nn2-c2cnnn2C)cn2cccc2c1=O CC1(C)CCCCCC1NC(C1CCC(NC(c2cc[n+]([O-])cc2)=O)O1)=O Cc1cnccc1C(N1CC(CF)(NC(C2COC(=O)C2)=O)C1)=O C=CCC(CC)C(=O)N(CCOCCCN(C(=O)C(C)C)C)CCO N1(C(COC2(C)CCC2)=O)CC2CC(C(=O)NCCOC3CC3)CC(C2)C1 C1(CNCC2CCCN(C(C)=O)C2)Cc2ccccc2C1=O CC1CCCN(C(=O)CN2CCC(C)(C)C2)C1CNC(=O)CCc1cn(C)cn1 c1(C(C(=O)NC(c2occc2Br)C)N(C)CC2CCCO2)ccccc1F c1(CC(=O)NC(CNC(C(C)OC)=O)C2CCC2)ccsc1Cl O(NC(=O)CN(C(=O)CC)CCN(C1CCCO1)C)CCC CN(CCCC(=O)N1CC(CC(N2CCOC(C)(C)C2)=O)C2(CC2)C1)N=O CC1CN(C(=O)C(N2CCC(C(F)(F)F)(CN)C2)=O)C(C)C1C c1(C(C(C)NC(c2c[nH]c(C(=O)O)c2)=O)C)ccc(C(F)(F)F)cc1 c1(NC(C(c2ccco2)OC)=O)ccc(OC2CCCC2)nc1 C1(N(C(c2ccc(F)cc2)C(=O)NCC(F)F)C2CC2)CCS(=O)(=O)C1 C(=O)(CCCC(F)F)NC(CNC(C1CCN(C)C1)=O)C1CC1 CCCCCC(C)(C)C(=O)N(CCCN(C)C(C1CC(=O)N(OC)C1)=O)C CC1CN(C(C2CCC(F)CC2)=O)C(C)CN1C(=O)CCc1ccccc1C#N CCC(CC(=O)N1CCC(CNC(=O)Cc2cnc[nH]2)(COC)CC1)C(C)(C)C N1(C(=O)C2=CCOC2)CCN(C(c2ccc(-c3cccs3)o2)=O)C(CCCCl)C1 C1(C(C(=O)NCC(CNC(C2(CC)CCCO2)=O)(C)C)O)CCCCCC1 N1(C(C2C(C)CCC2)=O)CCC2(CCOCC2)C(NC(c2cn[nH]c2)=O)C1 N1(C(c2c(C)nn(C)c2C)=O)CCC(N=c2ccnc(C(C)(C)C)[nH]2)C1 n1(CC)c(C)cc(C(=O)NCCCC2CCCCN2C(=O)C2=CCC2)c1C c1(-c2ccc(SC(C)C(=O)N3CCCC3)s2)ccc(F)cc1.C12CCCN1C2=O Cc1cnc(C(=O)NC2CCCN(C(C3CN4CCC3CC4)=O)C2C)c(F)c1 C1(NC(c2cnn(C)c2Cl)=O)CN(C(C2CC(=O)N(CC3CC3)C2)=O)CC1(C)C C1(NC(C2(CCCC)CC2)=O)CC2CC(NC(c3n[nH]c(CC)c3C)=O)C1C2 C1(C(=O)OC)(C(=O)NCC2CCCC2NC(C2(F)CCOC2)=O)CC(=O)C1 C1(C(=O)NCC(C)(C(C)C)NC(c2c(C)cc(C)nc2)=O)CC2(C1)CC(C)(C)C2 C1(N(C(=O)C=C(Cl)Cl)CCF)CCCN(C(C2CC3CCC2O3)=O)C1 C1(CNC(C(C=C)O)=O)CCN(C(c2nn(-c3ccccc3)cc2C)=O)C1(C)C c1(NC(C2CC2NCc2ccc(F)s2)=O)ccc2sc(Cl)nc2c1 C1(=O)C(C)(C)C(=O)N2CC(C2)OC2CCN1CC2.C(F)(C(=O)OC(C)(C)C)=CC C1(CC)CN(C(=O)C(C2CCC2)NC(=O)COCC2CCC2)CC1O N1(C(C(CCCC)NC(=O)COc2ccsc2)=O)CC(=O)NC2(CC2)C1 N1(C(c2cncc(O)c2Cl)=O)CCCC(C2CN(C(=O)C(O)C(F)F)C2)C1 CCCC(C)(C)C(=O)NC1CC(F)CN(C(=O)Cc2cccc(C(N)=O)c2)C1 CCC1=NOC(C(=O)NC2(C)CCN(C(c3nnn(C(C)C)c3C)=O)C2)C1 CCCC(C)(O)C(=O)N1CCC(C)(NC(=O)C(c2cc(F)cc(F)c2)C)C1 c1(COC)nc(Cl)cc(=NC2CC(NC(C3Cc4ccccc4C3)=O)C2)[nH]1 C(=O)(C1=CC2(CCOCC2)C1)NCC1(F)CC(NC(C2C(C(C)C)C2)=O)C1 c1(C(=O)NCCCN(C(C(C=CCCC)O)=O)C)cc2c(Cl)nccc2s1 N1(C(c2scc(C(C)C)n2)=O)CCC(CCN(C)C(C2C(C)CC2C)=O)CC1 N1(C(C(c2cc(C)sc2)(C)C)=O)CC2CC(NC(C3CCOC3(C)C)=O)CC1C2 n1(CC)cc(C(=O)NC(C)C=CC(=O)NCC(F)(F)CC2CC2)nn1 Cc1cccc(C)c1C(=O)NC1C=CC(C(=O)NCCCCc2ccccc2)C1 C#Cc1ccc(C)c(NC(=O)C(COC)NC(c2ccn3ccnc3c2)=O)c1 c1(CCC(=O)OC(F)F)c(Cl)cccc1F.CC1C(=O)N1 Cc1cccc(CC(=O)NCc2cc(C(N3CCCC3CN(C)C)=O)co2)c1 C1(CCC2N(C(c3nc(C)[nH]n3)=O)CCC2)CCN(C(=O)CC2CC2C)CC1 c1(C(=O)NC(C)CN(C(=O)CN2CCCCC2)C)cccc(SCC2CC2)c1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N2c1cc(C(F)(F)F)nc(Cl)n1 C(C(C)(COC)C(=O)N1CCCC1CNC(C1CC1c1cccs1)=O)OC c1(C(N2C(C(N3CCOC4CC34)=O)CC(O)C2)=O)[nH]nc2ncccc12 CC1CCN(C(=O)N(C)Cc2ncnn2C)c2ccccc21 C1(C(=O)NC(C2CCN(C(C3(C)CCCC3)=O)C2)C)CCC1(C)C C1(NC(CCC(=O)NC)=O)CCCC12CN(C(C1CC3(C1)CC3F)=O)C2 N1(C(C2(C(C)C)COC2)=O)CC(CCO)(NC(=O)CSc2cccs2)C1 C12(NC(c3c(C)cc(CC)o3)=O)CCCC1N(C(c1ccc(Cl)cc1C)=O)CC2 C12(C(N(C)CC3CN(C(C4OCC4(C)C)=O)CCO3)=O)CCC(CC1)CC2 CC1(C)CCCC(CC(N2CCC(O)(CCNC(=O)Cn3cnnc3O)C2)=O)C1 c12cc3c(ncnc3s1)[nH]2.c1(C(=O)NCC(CC)OCC)coc(C(C)(C)C)n1 n1(CCC)cc(C(=O)NCC2(CN(C(=O)CC(C)OC)C)CC2)c(C)n1 c1(CN2CC(C(C)NC(=O)C=Cc3ccccc3Cl)C2)c(Cl)cccc1B(O)O Nc1cc(F)c(C2CC2N2CC(=O)N(CC(=O)Nc3ccc(F)cc3F)C2=O)c(F)c1 N1(C(C(CC=CC)C)=O)CC(CC(=O)NCC(C)(O)CSC)CC1(C)C C=Cc1ccc(C(=O)NC2CCN(C(=O)C(C)C3CCC3)C(C)C2)cc1 C1(NC(CC(C)CN(C)C)=O)CN(C(c2cnc(NC3CC3)s2)=O)C2CCCC12 CC(CC(=O)N1CC2CN(C(c3nc(Cl)sc3C3CC3)=O)CCC12)C(F)(F)F CC1(O)CCN(C(C2(c3cn(CC4CCC(=O)O4)nn3)CCCCC2)=O)C1 C(=O)(C1=CCS(=O)(=O)C1)NC1CCC(F)(CNC(C2(C)CCCCCC2)=O)C1 C(CCC(C)C)(C(=O)O)NC(C(c1cccc(-c2nn[nH]n2)c1)OC)=O C1(C(N2CC(CC(=O)Nc3ccc([N+](=O)[O-])s3)(OC)C2)=O)CCCCC1(C)C c1(C(N2C(C)CN(C(C3CCCNC(=O)C3)=O)CC2)=O)nc2cccnc2s1 O=C(C1=CCCN(C(=O)CCCCCF)C1)NCC1CC1(Cl)Cl N1(C(CC(CC)C)=O)CC2(CCOCC2)C1Cn1cc(-c2c(Cl)cccc2Cl)nn1 c1(OCCOC)ccc(C2CCN(Cc3cccc(C#N)n3)C2)cc1OC(C)C C1(NCCC(=O)NCC=CCNC(Cc2c(CC)con2)=O)CCN(C)CC1 Cc1nn(CC(N2CCN(c3ncc(O)cn3)CC2)=O)c(=O)o1 c1(NC)ccc(F)cc1C(=O)NCCCN(CCO)C(c1coc(Cl)c1)=O C1(NC(c2c(C)cccn2)=O)C(CNC(c2cnoc2C)=O)CCC12CCC2 C1(C(=O)NCCN(C(C(C)OCCOC)=O)CC2CCCC2)CCCCC(=O)C1 C1(NC(CC(=O)NC2CC2)=O)CN(C(=O)C=Cc2ccsc2)CC12CCOCC2 C1(C(=O)NCC2(F)CC(CNC(c3nnsc3C)=O)C2)(OC)CCCOC1 c1(CN(CC(O)CN(C)C(C2CC2C(C)(C)O)=O)C)ccccc1 c1(SC)ccccc1C(=O)NC(c1nc(C)cn1C)c1ccccc1Cl c1(C(=O)NC2CC(C)(CNC(=O)C=Cc3cncs3)C2)ccnc2[nH]cnc12 c1(C(=O)NCCN(C(c2ccc(CN(C)C)[nH]2)=O)CC)ccc(Cl)c(C)c1 N1(C(C(C2(O)CN(C(CC(C)n3ccnc3)=O)C2)F)=O)CCC(C2=NOCC2)C1 C=CCCN=C(NCCc1cc(C)cc(Br)c1)NC(C)CC(F)(F)F N1(C(c2cc(C)c(C)o2)=O)CC(C2CCN(C(C3CCOC3(C)C)=O)CC2)C1 C1(C(=O)NCCC(CCC)C)CCN(C(=O)C=C(C)c2ccco2)C1(C)C c1(C(=O)NC(C)C(=O)N(CCCNC(C2C(Cl)(Cl)C23CC3)=O)C)ccccc1Cl N1(C(CCOCC)=O)CC(NC(c2nscc2C)=O)C(n2ccnn2)C1 CCCC(C(=O)N1CCCCC1CNC(=O)C(C(C)CC)OC)S(N)(=O)=O CC1CN(C(=O)C=Cc2cnc[nH]2)CC1NC(=O)CCOc1cccc(F)c1 Cn1ccc(-c2cn(CC(c3ccccc3)O)nn2)n1 N(C)(S(=O)(=O)N(C)C)CC(=O)NC1CCC(CNC(CN(CCC#C)C)=O)C1 c1(C(=O)NC(C)CCNC(=O)C(c2ccccc2F)O)ccc(P(C)(C)=O)cn1 CC(=Cn1ccnn1)C(=O)NCCCCN(C)C(C1CCC(F)(F)CC1)=O C1(C(=O)NCC(C)CNC(=O)COc2ccsn2)CCc2nn(C)cc2C1 N1(C(C(CCC)=CCC)=O)C2CCC1(CNC(c1cnc(O)s1)=O)CC2 CC(C)C(CCN(C(=O)CCc1cc[nH]n1)C)NC(C1(O)CCCC1)=O C1(CNC(C(COC)(C)C)=O)CN(c2nccc(C#N)n2)CCCO1 C(=O)(C(O)C(F)(F)F)NCc1nc(CNC(c2ccc(F)c(Cl)c2)=O)sc1 N1(C(C2C(CC)N(C(c3ccc(F)cc3)=O)CC2)=O)CC(OC)CC(C)C1 C1(NC(C2(N(C(c3ccc(C)cc3)=O)C)CC2)=O)CCCCCC1C Cc1ccc(C(C)(C)C(=O)NCC2CN(C(=O)C3=CCC3)C3CC23)cc1 c1(C(N(C(C(N2CCCC(OC)CC2)=O)C)C2CC2)=O)c[nH]c2cnccc12 Cc1ccc(S(=O)(=O)N2CCC(C(=O)Nc3nc4ccsc4s3)C(O)C2)c(C)c1 c1(CCNC(C2CC2F)=O)ccc(CNC(C2CC(F)C2)=O)cc1 C(CCF)(C(=O)NCCCc1nccs1)NC(C1C(C)OCC1)=O c1(C(N2CC=CC(NC(c3cc(C(C)=O)c(C)o3)=O)C2)=O)nnc(O)cc1O C(=O)(C(=O)NCCF)N(CC(C)C)CCN(CCC)CCC1CC1 c1(C(N2CC(O)(CC)C2)=O)ccc(CNC(=O)CSc2ccccc2)cc1 C1(C(N2CCC(COC)(CNC(=O)C(C)C3CC3)CC2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NCc2nnc(C)s2)CC(C)CN(C(C2C=CC=CC=C2)=O)C1 C=CCN(OC)C(=O)C12CCC(NC(=O)CNC(=O)CC(C)C)(CC1)C2 C1(CNC(C(CC(=C)C)C)=O)CC12CCN(C(=O)C(=O)NC(C)C)CC2 c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(C2COC(=O)O2)=O)C1 C1(C(=O)NC(CNC(C=C2CCC(C)CC2)=O)(C)C2CC2)COC2(CCC2)CO1 N1(C(c2c(C)cnnc2)=O)Cc2nccn2CC(NC(C2(C)CCCN2C)=O)C1 c1(SCCC)cccc(C(=O)NC2CN(C(=O)C(C)(O)CC)CC2SC)c1 S(=O)(=O)(c1cscc1F)N(C)C.c12ccccc1NC(=O)C2 c1(OC)c(C(=O)NC2(CO)CC(NC(C=CC)=O)C2)cnn1C.C1(N)CCC(O)CC1 C1(CC(=O)N(CCCCC=C)C)CC2(CC2)CN1C(=O)CSC(C)(C)C c1(OCCC(=O)N(CCNC(C(CC)COC)=O)C(C)C)ccc(Cl)cc1Cl C=CCCC(C(=O)NC(C)C(C)NC(c1cnc(S)n1C)=O)c1ccccc1 C1(N(C(=O)CS(N)(=O)=O)C)CN(C(=O)CNC(C2CCOCC2)=O)CC1(C)C C(=O)(CCC(F)F)NC(CNC(C(n1ccc(C(F)(F)F)n1)C)=O)CO [N-]=[N+]=NC1CC(C(=O)NC2CC3CCC2O3)N(C(c2ccc(C#N)cc2)=O)C1 Cc1ccc(-c2ccc(C(=O)NC3CC(F)(CNC(c4ccsn4)=O)C3)s2)s1 C1(CO)CN(CCC2CCCC2(F)F)CC12COC2 c1(CC(N2CCC(n3cc(CN(C)C)nn3)C(O)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(C1=Cc2ccccc2C1O)NC1C(C)(C(C)C)C1 C1(C(=O)NCC(C)Cc2cn[nH]c2)CCN(C(C2CCCCC2)=O)C1(C)C c1(OC)c(C(c2nnnn2CCC2(C)CC2)NCC(C)OC)cccc1Cl C1(c2nc(C(C)C)on2)CC2CC(C1)N(C(C1CC1c1ccc(Cl)s1)=O)C2 C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)CSc2nnnn2C)CC1C C#CCC(O)C(=O)N(C)CC1CCCC1NC(=O)C(C1CCOCC1)F N1(C(CC(c2ccc(F)cc2)C)=O)CC2CC2(CNC(c2ccsc2C#N)=O)C1 C1(CC)CN(C(=O)C(c2ccccc2F)(C)C)CCC1NC(C1(Br)CC1)=O C1(NC(=O)CC2CC2)CC(CNC(C2CCN(Cc3nncs3)C2)=O)C(O)C1 Cc1ccc(C(=O)NC2CCCC2NC(C2(C(C)(F)F)CC2)=O)c(Cl)c1.C1(C)CC1 N1(C(C(CCOC)C)=O)CCN(C(c2cn(CCCF)nn2)=O)C(C)C1 Cc1cc(C(c2nnnn2C)NC2CN(c3ccccc3)C2=O)sc1Br C1(C(=O)NCC(C)S(N)(=O)=O)(NC(c2cc(COC)no2)=O)CCC(C)(C)C1 c1(OC)ccc(Cl)c(C(=O)NCCC2CCCCN2C(=O)C(C)n2cccc2)c1 N1(C(C(CC(C)C)O)=O)CCCCCC(NC(c2ccc3ncnn3c2)=O)C1 c1(NCC(=C)Cl)cc(=NCc2nc(C)c(-c3ccccc3)o2)[nH]cn1 c1(C(N2CC(F)CC(NC(C(C=C=C)C)=O)C2)=O)ccc2cc(O)ccc2n1 CCCCCC(O)C(=O)N(C(C)(C)CC(=O)NCC1CC(F)(F)CO1)C C1(COC)(CNC(=O)Cc2cc(C)on2)CCN(C(c2ccc(SC)s2)=O)C1 N1(C(C(C)=CC)=O)CCC(C(C)C(=O)NCC2CN3CCC2C3)CC1 C=C=CC(C)C(=O)NCC(C)N(C)C(c1c(C(F)(F)F)coc1CC)=O c1(CC(=O)NC2CN(C(=O)OC(C)(C)C)CC(F)C2)c[nH]c2ccc(Br)cc12 C1(CNC(c2c(CC)c[nH]n2)=O)CC12CCN(C(=O)CC1CC(C)(C)C1)CC2 C1(CCC)CC(C(=O)N(C)CCNC(c2nc(C)n(C)n2)=O)CCO1 N1(C(C(CC2CCCC2)NC(C(CC=C)(F)F)=O)=O)CCC2(CC1)CN(C)C2 C1(CNC(c2cccc(CNC(C3CC4C=CC3C4)=O)n2)=O)CCC(CO)CC1 C1(NC(C(C)SCC2CCCO2)=O)CC2(C1)CC(NC(C1CNC(=O)N1)=O)C2 C(=O)(C(CC(C)C)CC(C)C)NCCN(C(C)C)C(c1cc(F)ccc1NC)=O c1(C(N2CC(=C(CNC(C(COCC)N=[N+]=[N-])=O)F)C2)=O)nc(C)c(C)[nH]c1=O N1(C(C(C2CN(C(=O)C(C)(C)Cl)C2)OCC)=O)CCCC1C(C1CC1)OC c1(C(N(CCCNC(c2cc(C(CC)C)no2)=O)C2CC2)=O)cc(O)ccc1C S(=O)(=O)(c1cccc(Cl)c1)N1CC(C(N2CCCC(F)C2)=O)OCC1 C12(CNC(c3ncc(C)nc3)=O)CCCC1CN(C(=O)C(C)C1CC1)C2 C#CC1(C(=O)NCCc2cccnc2)CCN(C(=O)CC(CC)SC)C1 N1(C(C2(CC(N)=O)CC2)=O)CC(CNC(=O)CC2CC(N(C)C)C2)C(O)C1 c1(C(N(CC(CC)NC(C2CC2c2ccsc2)=O)C)=O)ccc(F)cc1[N+](=O)[O-] C1(NC(C2(CC=C)CC2)=O)CCC2(CCN(C(c3cc(C(C)=O)oc3C)=O)C2)C1 c1(CC)conc1CC(N1CCC(Cc2cn(CCCN3CCCC3)nn2)C1)=O N1(C(C(=O)Nc2ccc(C)cc2)=O)CC(C)N(C(c2cccc(Cl)n2)=O)CC1C C1(CC)CN(C(c2ccnc(OCCO)c2)=O)CCC1NC(=O)CC1CN(CC)C1 C(C(C)N=c1[nH]c(Cl)nc(C)c1F)NC(Cc1ccc(C)cc1Cl)=O c1(C(=O)NCCCCCn2cc(CCN(C)C)nn2)n[nH]nc1OCC(F)F N1(C(c2cc(CC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)COC(C)(C)C C(CC#CC)(C(=O)N(C)Cc1cccnc1)NC(C(C=C)O)=O c1(CCC)ccc(C(=O)NC2COCC2CNC(=O)C(C)(O)CC)cc1[N+](=O)[O-] C1(C(C)C)C(C(=O)N(C)CCN(C)C)CCN1C(=O)C=C1CCC(C)CC1 CCC(CC(=O)N1CCOC(CCCNC(=O)C=CCn2cncn2)C1)C(C)C C1(C(N2C(CC)CC(C)C2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C N1(C(C2(C3CC3)CN(C(C3CCCC(=O)C3)=O)C2)=O)CC2CCC(C1)C2O N1(C(CC(C=C)CCC)=O)CCCCC2(C1)CN(C(=O)CC(F)(F)F)C2 C1(C(=O)NCC(COC)NC(=O)C(O)C2CCC2)CCCCN1C c1(COC)cc(C(N2CC(O)(C(C)NC(=O)CCCc3csc(=N)[nH]3)C2)=O)n[nH]1 Cc1cccc(NCc2cn(CC(=O)NC(c3cccnc3)CO)nn2)c1C c1(C(N2CC3CN(C(C4(n5ccnn5)CC4)=O)CC3C2)=O)cc(Cl)c(F)cc1Cl N1(C(C2CC(C)(C)C2)=O)CCC2(CCCN(C(=O)Cc3ccc(F)c(F)c3)C2)C1 c1(C(=O)NCCCCN(C(=O)C(C)(C)CN(C)C)C)c(F)ccc(F)c1O CCC(C)C(C(=O)NCCCCCO)NC(c1ccc(=N)[nH]n1)=O c1(C(N(CC(C)CNC(=O)CC2COC(=O)C2)C)=O)ccnc2[nH]cnc12 c1(C(=O)NCCOC2CN(C(C3CC34CCCC4)=O)C2)ccccc1Br C(=O)(C(CO)NC(c1cc(C)cs1)=O)NC1CC(SCC)C1 C1(C(=O)NC2CCCC(NC(C(CC=C)(F)F)=O)C2)COc2ccc(F)cc2C1 c1(OC)cccc(NC(=O)C(c2nocc2Br)N(C)C(C2CC2)C2CC2)c1 Cc1ccc(NC(c2cnn(CC(c3ccc(C)o3)C)c2)c2nnnn2C)cc1 CC1(C(=O)NCC(O)CNC(=O)C2=CCC2)COCCO1 c1(CC)cc(C(=O)NCC2CCCN(C(c3cnc(C(C)O)s3)=O)C2)nn1C C(=O)(C1=CCCSC1)N1CCC(CCCCCNC(Cc2c(C)ocn2)=O)CC1 N1(C(COCC)=O)CC2CCCC(C1)N2C(C1CC12CCOCC2)=O c12ncc3c(n1)CC1CCC3N1C(=O)C2.C1(C(C)(C)C)CCC(C(F)(F)F)CC1 C12(CCC(=O)NC3(CNC(=O)CC4CCOC4=O)CCCC3)CCC(CC1)C2 ClCCCN=C(NCC1CCCO1)NCC(c1ccc[nH]1)OC1CCC1 c1(C(=O)NCCN(C)C(c2ccc3nnnn3c2)=O)nc2n(c1Br)CCC2 c1(OCC(C)C)ccc(C(N2CC(O)(C(C)NC(C3(C)CSC3)=O)C2)=O)cc1 C1(NC(c2snc(C(CC(C)(C)C)(C)C)n2)=O)(CO)CCc2ccccc2C1 C1(C(N2CCC(N(C(=O)CN3CCCCC3)CC)C2)=O)CCS(=O)(=O)C1 C(C=CC(=O)N(CC(N1CCCC1)C)C(C1CCOC1)=O)(CC)=CC C1(N(C(CC(C)O)=O)C2CC2)CCNCCC1C N1(C(CCC(=O)OC)=O)CCC2(CC1)CC(C)N(C(=O)Cn1ccnn1)C2 C(CC(F)(F)Cn1cc(CO)nn1)N(C)C(C)=O.C=CCCCN C1(CNC(C(C)NC(CC)=O)=O)CC2CN(C(=O)C=C(C)C(F)F)CC12 CC1CCC1N=c1nc2scnc2c(N2CCN(C(=O)COC(F)F)CC2)[nH]1 Cc1n[nH]c2cnc(C(=O)NCC3CCN(C(C4CC5CCCCC45)=O)C3)cc12 n1(CC)ccnc1C(N1CC(O)(CNC(=O)CC2CCOC2C)C1)=O S(=O)(=O)(c1ccc(Cl)cc1Cl)N1C2CN(C(C3C(C)C3)=O)C(C2)C1 C(C)(C(O)C(=O)OC)N1CC2C(C(=O)OC)(C2)C1 N1(C(c2c(CC=C)cccc2)=O)CCCC2C1CCN2C(C1CC(C)C1)=O c1(C(=O)NOCC)ccccc1Sc1ccccc1OCC(C)C#N n1(CC(=C)C)c(N2CCC(Oc3cncc(Cl)n3)CC2)nnc1CO C1(OCc2nc(-c3ccc(OC)nc3)nn2-c2ccnn2C)CCCC(F)(F)C1 c1(C(CCO)NC(=O)NC(C)C(C)(C)C#N)ccc2c(c1)OCCO2 C1(CNC(CC(CCC)O)=O)CCN(C(=O)Cn2ccnc2C)C12CCC2 C1(NC(C=C(C)Cl)=O)CN(C(c2ccn3ccnc3n2)=O)CCC1(C)C C(=O)(C1=C(Cl)CCCC1)N1C(CCCC(=O)NC2(C(=O)OC)CCCCC2)CCC1 Cc1occ(C(F)(F)F)c1C(N1CCC1C(=O)NC(c1cnn(C)c1)C)=O c1(C(=O)NC2(CC)CCN(C(c3cc(C)n(C)c3)=O)CC2)cc(F)c(C)cc1F c1(C(C)C)nccc(=NC(C)C2CCCCN2C(c2ccn(C3CC3)n2)=O)[nH]1 Cc1nc(C2CC2)[nH]c1C(=O)N(CC(F)F)Cc1ccccc1 N1(C(c2nc(C)[nH]n2)=O)CCCC(C2CCCCN2C(=O)CC2CCN(C)C2)C1 C1(C(N(C)Cc2ccc(C)cn2)=O)CC2CCCC2N1C(=O)C=CC1CC1 C(CCC(C)(C)C(=O)N1CC2CCC(C1)N2C)NC(C1N(CC)CCC1)=O C(=O)(C1=CC2CCC(C1)C2)NCC12OCC(CNC(C(N=S(C)(C)=O)=O)=O)(C1)C2 Cc1ccn(CC(=O)NCC2(CNC(c3cncc(Cl)c3Cl)=O)CC2)c(=O)c1 Cc1cn2c(C(=O)NCC(C)(O)CNC(C3CC3C)=O)cnc2s1 N1(C(c2n(C)cc(NC(c3cncc(C)n3)=O)n2)=O)CC2COCC2C1 N1(C(c2ccc(-c3ccc(C)o3)s2)=O)CC=CC(NC(=O)C(F)F)C1 c1(OC)ccc2[nH]c(=NCCCCCCCO)nc(N3CCC(CC#N)C3)c2c1 N1(C(CCCOC)=O)CCCC2C1CCN2C(C1CC2CCN(C1)C2=O)=O C=C(C)C1OCCC1C(N1CCC(CCC(N2CCCC2C(O)CO)=O)C1)=O c1(C(=O)NC(C)C(C)C(=O)N(C)CCc2cccs2)cc2ncccc2[nH]1 Cc1cccc2cc(C(=O)NC3C4CC3N(C(=O)CC3CCCCC3O)C4)oc12 N1(C(c2cc(SC)oc2)=O)CCCC(CNC(=O)C(c2ccccc2)F)C1 c1(C(=O)NCC(C)(C)NC(C(n2ncc(C)c2)C)=O)c[nH]nc1[N+](=O)[O-] Cc1ccc(Cl)c(OCC(N2CC3CC3(CNC(C3(CF)COC3)=O)C2)=O)c1 C(=O)(CCC1=CCCCC1)N1CCC(NC(C2(C)CS(=O)(=O)C2)=O)C(F)C1 c1(CC=CC(=O)NCc2csc(CNC(c3ccsn3)=O)n2)ccc(Cl)cn1 c1(C(=O)OCC)cc(Cl)c(Cl)c(CN2CC(CC)CC2=O)c1Cl c1(OC)ccc(C(N2CCCCC2C2(NC(=O)CC34CCCC3C4)CC2)=O)nc1 C1(CC(=O)NC(CSC)CO)CN(C(C2(OC(C)=O)CCOC2)=O)CC12CC2 Cc1cc(Br)cc(C(N2CCN(C(=O)C=Cc3cn[nH]c3)C(C)C2)=O)c1F Cc1cc(C(=O)NC2CN(C(=O)CC3CC3)CC2n2ccnn2)sc1C(=O)O N1(C(C(CC)OCC)=O)CC2(CCC(NC(=O)C(=Cc3c[nH]cn3)F)CC2)C1 c1(CNC(C2C(C(C)C)OCC2)=O)ncc(C(=O)N(CCC2CC2)CC2CC2)cn1 c1(C(=O)NCC2(O)CCN(C(C(C)(C)C3CCC3)=O)C2)ccn2ccnc2n1 c1(C(N(C2CCC(NC(CCCC)=O)C2)C)=O)ncn2c1CCC2 C1(N(C(C(C2CCC2)OC)=O)C)CCCCN(C(c2ccc(C(N)=O)cn2)=O)C1 C1(CC(=O)NCc2c(C(N(c3cccc(Cl)c3)C)=O)n(C)nc2)CCCC2CC12 C(C(C)C)(C(=O)N(CC(C1CC1)N(C)C(C)=O)C)NC(CNC(=O)OCC)=O c1(-c2c(C(=O)O)c[nH]n2)cc(Cl)cc2c1OCC2 CC1CC(NC(=O)Cc2cncc(F)c2)CN1C(=O)COC1CC=CC1 c1(C(N2C(CCOC)CN(C(c3cc(Cl)no3)=O)CC2)=O)cc(C)c(C)cc1C c1(C(N2CC(C(C)(C)O)(CNC(CSC)=O)C2)=O)ccc(OC(F)F)c(Cl)c1 C=CC(CC)CC(=O)NCCCNC(c1ccc(CC)nc1C)=O c1(CC)cc(C(=O)NCCCN(C(=O)CCOC)CCO)c2ccccc2n1 C12(C(=O)NC3CN(C(CNC(=O)CC(F)(F)F)=O)CC3O)CCCC(C1)OC2 CC#CCCCC(=O)NCC(C)(C)C(=O)N(CC(=O)NC)CC c1(C(N2CC(C3N(C(CC=C)=O)CCC3)(O)C2)=O)cc([N+](=O)[O-])nn1C C(=O)(CCCC(=O)N1CCC(NC(=O)CC(c2ccccc2C)C)C1C)OCC N1(C(c2scc(C)c2)=O)CC(NC(c2cc3ccsc3s2)=O)CC12CCOCC2 C1(CNC(CC)=O)CN(C(c2cccnc2OC(C)C)=O)CC1C CC1=C(C)CC(C(=O)NCc2cc(C)c(C(=O)NCc3cccnc3C)o2)CC1 C12(C(C(=O)N(C3(C(=O)NCC4(CCCC)CC4)CC3)C)C)CCC(CC1)C2 N1(C(c2c(C)c(F)ccc2)=O)CC(NC(c2ccnnc2S)=O)CC2(CCC2)C1 N1(C(C2C(C)(C)CO2)=O)CC2CC1CN2C(c1cnc(O)o1)=O C12(C(N3CC(O)(CN(C(=O)CC4C=CCC4)C)C3)=O)CC3CC(CC(C3)C1)C2 N1(C(C2(C(C)(C)O)CC2)=O)CCC(C)(C)C(NC(c2ccc(NC=O)cc2)=O)C1 CCCCCC(=O)N(CCC(=O)NCN1CCC1)CC.OC c1(C(N2CCC(CN(C(c3c(C)scc3)=O)C)C2)=O)ccc2c(c1)CC2 CC1(C)CC(C(=O)NC2CCC(CNC(C3CC4CC4C3)=O)CC2)(CO)C1 C(=O)(CCC(C)O)NC(CNC(CCOCCCOC)=O)C(C)C c1(OC)ccc(C(C)C(N2CC(NC(=O)Cc3cnc(C)o3)C(C)C2)=O)c(C)c1 Cc1ncc(C(=O)NC(Cc2ccccc2)CCNC(=O)C(C)(C)F)n1C C1(C(N2C3C(C(N4CCSCC4)=O)CC(CC3)C2)=O)C2Sc3ccccc3C12 N1(C(C(CC)c2ccco2)=O)CCC2(CCCN2C(=O)CCNC(N)=O)C1 N1(C(C2C(C)=CCC=C2)=O)CCCCC(N=c2nc[nH]cc2C#N)C1 N1C(N2CCC(CC3CC3)C2)=NC1.C=CC(C)N(C)C(=O)OC C1(NC(c2n(CCCC)ncc2)=O)CC(O)CN(C(=O)CC2CCC=CCC2)C1 N1(C(C(CC)(F)F)=O)CCCC(F)(C(NC(=O)C(COC(C)(C)C)N(C)C)N)C1.OC N1(C(c2c(OC)nc(C)cn2)=O)CC2(CCCN(C(=O)CN(C3CCC3)C)C2)C1 c1(C(C)C)cc(C(=O)NCC(CO)NC(c2sccc2OC(F)F)=O)n[nH]1 C1(NC(c2nc(CCC)oc2)=O)CC2CC(C1)N(C(C1(C)CC(O)CN1C)=O)C2 C1(NC(C(C)=C2CC2)=O)CC1C1CCCN(C(c2c[nH]cc2-c2ccccc2)=O)C1 N1(C(c2csc(CN3CCCC3CO)n2)=O)CCC(O)C1.C12(CO)CCN(CC1)C2 C1(CC)(Nc2ncnc(Cl)c2CO)CCN(C(c2cc(=O)cc[nH]2)=O)CC1 CCC(C)(COC)C(=O)NN1CCCC1C(=O)NCCC1CC(C)C1 C1(N2CCN(C(=O)OC)CC2)CCCC12CN(C(=O)C(C)Oc1ccccc1)C2 N1(C(c2c(SC)cccn2)=O)CCC(C)C(NC(=O)CC(C)(C)CC)C1C Cc1cnc(C(=O)NC2CCCC(NC(C3CCC(C(N)=O)CC3)=O)C2)cn1 N1(C(N2CC(C)C(C(=O)OC(C)(C)C)C2)=O)CC(C)C(F)(F)C1 C=CCC(CC(F)F)NC(C1CN(C(=O)CC2(OC)CCC2)CC1C)=O CC(C)CCC(C(=O)NC(C)C(=O)N1CCCC1)NC(=O)CCCN(C)C N1(C(C(CO)OC)=O)CCOC(CNC(=O)C(N2CCC(O)CC2)C)C1 N1(C(C(C=C)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC(C)(F)C1 C1(NC(CCC(=O)OC)=O)CCC(C)N(C(C2CC(O)(C(F)(F)F)C2)=O)C1 CC1CN(C(=O)C(C2(O)CCCC2)F)CC1NC(=O)Cn1cc(C#N)cn1 Cc1cccc(CNC(=O)C(C)(C2CC2)N(C)C(c2cncc(CO)c2)=O)c1F N1(C(C2CC2(C)C)C(=O)Nc2c(C)cccc2)CC23CCCC2(COC3)C1 C(=O)(C1CCc2cccc(OC)c21)NC(CC=C)CNC(=O)Cn1cc(Cl)cn1 CC1(C)CC(C(=O)NC2CNC(=O)C2)CCN1C(=O)C(F)=CC1CC1 Cc1[nH]cc(C(=O)NC2CN(C(=O)C(C)C3(O)CCC3)CC2(C)C)c(=O)c1Cl C1(C(N(C(CNC(c2occ(C)c2)=O)(C)C)C)=O)CC12CC(O)C2 C#CC1(C(=O)Nc2ccc(OC)nc2)CCN(C(=O)CC2CCC2)CC1 C(=O)(CCCCNC(C1CCCCN1C(c1ccc(F)s1)=O)=O)OCC N1(c2ccnc(Nc3c(C)ccc(Br)c3)n2)CCC2(CC1)CC(C1=CCCC1)=NO2 C1(C(=O)NCCN(C(C2(O)COC2)=O)C2CC2)CCCC1n1cccc1 Cc1ncc(N)cc1C(N1CCOC(CC(=O)NCc2n[nH]cc2[N+](=O)[O-])C1)=O c1(C(=O)NC2CCN(C(C(C(CC)O)(F)F)=O)C2)sc2cccc(F)c2c1Cl C1(NC(c2cnc(S)[nH]2)=O)CC2CC(C1)N(C(c1ncsc1Br)=O)C2 Cc1nccc(-n2cc(C3CC(NC(C4CC(F)(F)CS4)=O)C3)nn2)n1 C(=O)(CCCC(CC)NC(=O)C1=C(C)OCC1)N(C1CC(CC)C1)C c1(C(N(C)CC2N(C(CCCCC=CC)=O)CCC2)=O)cnc2cnn(C)c2c1 C1(C(=O)Nc2scc(C)n2)CC12CCN(c1ncnc(C)c1Br)C2 N1(Cc2cn(C)cc(Br)c2=O)CCCC(N=[N+]=[N-])CC1 C(=O)(C=C1SCC(=O)N1C)N1CC(NC(C(CC=CCC)C)=O)C(OC)C1 C12(C(N(C3CCC(F)(F)C3)C)=O)COCC1CN(C(=O)C(C)(C)C)C2 c1(N(CCC)CCNC(C2(C)CCC(=O)NC2)=O)ncc([N+](=O)[O-])cc1F CCCC(C)(C)C(=O)NCC1(O)CCCN(C(=O)CCc2ncccc2C)C1 C(=O)(C(=O)C(C)CC)NCCCNC(C(CSC)O)=O C1(OC)CC(CNC(=O)Cn2nnc(=O)[nH]2)N(C(=O)C=CC2CCOC2)C1 n1(CCCC)nc(-c2ccc(OC)cc2)nc1C1CC1c1ccccn1 c1(C(C)C(=O)NC(C)(C)CN(C(=O)CC2CCC23CCC3)C)c(F)cccc1F c1(NC(c2c(NC(c3c(C)scc3)=O)ccs2)=O)ncc(Br)nn1 C1(CNC(Cc2c(C)n(C)cn2)=O)CC2CCC1N2C(=O)CC=CC(C)(C)C C1(C(=O)NC(C2CCCCC2)C)C2CN(C(c3ccc(CO)cc3)=O)CC12 C(=O)(CCCCC(C)(C)C)NC1CC(CCNC(C(C)NC(=O)C2CC2)=O)C1 C1(CCC=C)(C(=O)NCC(O)CO)CN(C(=O)Cc2ccc(Cl)s2)C1 C(C1CCCC1)=C(C)C(=O)NC(C)C(=O)NC(C)Cc1nn[nH]n1 c1(CN(C(CN2CCC(CCCC)C2)=O)C)ccccc1Cl C1(NC(c2cc(C)nn2C)=O)CCN(C(c2sc(Cl)cc2Cl)=O)C(C)C1 N1(C(C(=O)NCCC=C)C(C)C2CCCCC2)CC2CCC1CC2CO N(C(=NCCCOCCN(C)C)NCC1(S(C)(=O)=O)CCCC1)CC1C(C)C1 N1(C(C2CCCCO2)=O)CC2CC1CN2Cc1nc(C2CC2)no1 Cc1nn(-c2ccccc2)cc1C(=O)NC12CC1CN(C(=O)Cc1cocn1)C2 C1(NC(c2ccc(C)cc2)=O)CCN(C(=O)CC#N)CC1(C)C c1(C(N(CCCNC(=O)C(C)c2cc[nH]n2)C(C)C)=O)cc(N)nc(Cl)c1 C1(NC(=O)NCC2C(C(N3CCN(C)CC3)C)C2)CCC(OC(F)F)CC1 CCC(C(=O)NCCC1CCN(C(c2[nH]nnc2C2CC2)=O)C1)c1cccnc1 C1(CNC(c2c(C)nns2)=O)CN(C(=O)CCc2nncs2)CC1O C(=O)(C(N=[N+]=[N-])C(C)C)N1CCC(CC)CC1C(=O)N(CC(F)F)C c1(C(N2CC(NC(c3cnc(CC)[nH]3)=O)C(C)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(NC(C2CCC(CNC(C(C)n3cnnn3)=O)CC2)=O)CN2CCC1(C)CC2 CC1(C)CCCC(C(=O)NCCC2(NC(c3cnc(O)o3)=O)CCC2)CC1 C1(C(=O)NCCC2CSCCN2C(=O)CCN2CCCC2=O)COC2COCC12 C(CC(=O)NCc1ccccc1OC(F)F)(C(F)(F)F)N1C(C)CCC1C c12nc(nc3c1COCC3)CN2C.c1(OC)ccc(N2CCCC2)cn1 c1(-c2c(C(=O)NC(CCC#C)(C)C)cccc2)ccc(Cl)c(Cl)c1 C1(Nc2ccc(CN(CC(N)=O)CCC)cc2)CCOC12CCOCC2 c1(C(=O)NCCC(C)NC(C2C(C#C)C2)=O)cnn(-c2nc(SC)ns2)c1 C1(C(N(C2CCN(C(=O)CC3(O)CCCOC3)C2)C)=O)CCC(C(C)(C)O)CC1 Cc1cc(N)c(F)c(C(=O)NC(CNC(C2CC23CC3)=O)C2CC2)c1F CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CC1(C)CNC(=O)C(c1ccccc1)F C1(C(N(CCn2cc(-c3ccc(C)nc3)nn2)C2CC2)=O)CCCC(C)(C)C1 c1(NC(C23CC(NC(C(C)Sc4ccccc4)=O)(C2)C3)=O)ccc(N)cc1Cl N1(C(C2C(=C)C2)=O)CC2CCC1CC2NC(=O)C(C)(C)CF CCCC(C(=O)NCCc1ccc(C)nc1)NC(=O)C(O)Cn1cncn1 C1(C(=O)NC2(COC)CN(C(c3cc[nH]c3C)=O)C2)Cc2cc(F)ccc2O1 C(=O)(C(CC)CC(C)C)N1C(C(=O)NCC(C#C)C(C)C)CSCC1 Cn1nc2c(c1C(N1CCC1CO)=O)CN(Cc1c(F)cc(OC)cc1F)CC2 CC1CCCN(C(=O)C=Cc2cn(C)nn2)C1C1N=N1.C1(=O)CN1.C1C=CCO1 c1(C(N(C)CC2CCN(C(C(CCC)OC)=O)C2)=O)cc(S(N)(=O)=O)cs1 CCCC(CC)CCC(=O)NC1CN(C(c2ccc(C#N)s2)=O)CC1O N1(C(C(CNC(CCCCC=C)=O)C(C)C)=O)CCC(C2CCC2)CC1 C1(CNC(C2CSCC(=O)N2)=O)CN(C(c2cocc2Br)=O)CCO1 C(=O)(CC1=NNC(=O)C1)NC(C1CCCN1C(c1ccc(=N)[nH]n1)=O)C Cc1cc(F)c(CNC(=O)C(=O)NCCC(C)C)cc1Br.C1(C)CCN1 C1(CCC(=O)OCC)CCN(C(=O)C(=O)N(C)Cc2c[nH]nc2OC)C1 C1(C(=O)NCc2ncc(C)o2)CC2(CCN(C(=O)C(N3CCNC3=O)C)C2)C1 c1(CNC2CC(N(C)C(c3c(Cl)ccc(N(C)C)n3)=O)C2)ccc2ccsc2c1 CC(=O)C(C)(C)CC(=O)NC1CS(=O)(=O)CC1Nc1cc(O)ncn1 c1(OC)ccc(F)c(C(=O)NCCCNC(C2CC(C#N)(OC)C2)=O)c1F c1(C(=O)NC2C(OC)COC2)oc(CNC(C2(CO)CCCC2)=O)nc1C C#CCC(C(=O)NCc1cnn(C)c1)NC(c1coc(C(C)C)n1)=O C1(C(N2CCCC(C)(O)C2)=O)CCC(C)(C)N(C(C2(F)CCOC2)=O)C1 CC(O)CCCCCC(=O)Nc1ccccc1CN1CNS(=O)(=O)CC1 C1(NC(c2cncnc2)=O)CN(Cc2ccc(-n3ccnc3)cc2)CC1O c1(C(=O)NCC2CN(C(c3c(C)onc3CO)=O)CC2C)c[nH]c(=N)nc1C N1(C(CCNC(=O)OC)=O)CCN(C(c2cc(O)nc(C)n2)=O)C(CO)C1 CC(C)CCCC(C)C(=O)N(C)CCC1CCN(C(C2COC(=O)N2)=O)CC1 C1(NC(=O)CCC2CCC2)CCCC2CN(C(=O)CNS(N)(=O)=O)CC12 CCCC(C)C(=O)N1CCC(F)(C(=O)NCC(c2ccc(O)cc2)O)C1 c1(OC)ccc(CC(N2CCC(C)(C(N3CCC(C)(O)C3)=O)CC2)=O)c(F)c1 C1(NC(C(CCN(C)C)O)=O)(CO)CCCN(C(=O)Cc2cccc(O)c2)C1 N1(C(CS(CCOC)(=O)=O)=O)CCCC2(CCC2NC(C2CCCC(CF)C2)=O)C1 C1(C(=O)NCc2cc(C(N(CC)CC)=O)no2)CCOC(C)C1 CC1CCN(C(C2CC(NCc3cc(Br)c(F)cc3F)C2)=O)CC1(F)F C1(NC(C(c2cccnc2F)(C)C)=O)CN(C(c2cc(C3CC3)cs2)=O)CC1F c1(OC)ccc(C(=O)NC2CC(F)CN(S(=O)(=O)CC3CCC3)C2)cc1F C1(NC(C(C)N2CCC2)=O)C(C)CCN(C(c2cscc2C(F)F)=O)C1C C(C1=CCCN(C(C2(F)CCCCCC2)=O)C1)NC(c1ncccc1C(F)F)=O C(CC(=O)NC1CCC(C(C)C)CC1)(C(C)C)NC(c1c(CCC)cccc1)=O C1(C)(C(N(C)CCOCCCNC(=O)CC23CCC(CC2)C3)=O)CCCS1(=O)=O C1(CNC(=O)C(O)C2CC2)COCCN1C(C1CCCC1Cc1ccccc1)=O C1(NC(=O)CCOCC(F)(F)F)CS(=O)(=O)CC1N=c1ccnc(C2CCC2)[nH]1 N1(C(c2c(NC)snc2C)=O)CC(NC(=O)CCc2ccccc2)CC(O)C1 C1(CNC(C2(CCOC)CC2)=O)CC(C(=O)N2CC(C(N)=O)C3(CC3)C2)=NO1 c1(C(=O)NC(C(C)C)C(C)NC(c2cnn(CCF)c2)=O)cccc2ccoc12 N1(C(CC2(C=C)CC2)=O)CC(CNC(c2nnc(S)n2C)=O)OC2(CCC2)C1 C(c1ccc(C#N)cc1)=CC(=O)NC1CCC(C)N(C(c2cccc(=O)o2)=O)C1 N1(C(C=C(C)CCc2ccccc2)=O)CC2OCC(NC(=O)C3=CCCS3)C2C1 CCC(O)C(C)(C)C(=O)N1CC(C(C(N2CCC(c3ncc[nH]3)C2)=O)OC)C1 c1(NC(C(c2cc(O)cc(Cl)c2)N2CCC(C(=O)NC)C2)=O)ccc(Cl)cc1F C1(NC(c2ccnc(OC)n2)=O)CC2CC1N(C(C1CCCN(C(N)=O)C1)=O)C2 c1(C(N2C(CNC(c3c(CC)noc3)=O)C(C)CC2)=O)cncc(S(N)(=O)=O)c1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CC(C)CN(C(c2cc(O)nc(Cl)c2)=O)CC1C C1(NC(C2CCOC2)=O)CCC(NC(=O)C(F)(F)COc2ccc(F)cc2)CC1 C12(C(N3C(CNC(c4ncsc4C4CC4)=O)CCCC3)=O)CCCN(CCC1)C2 c1(NC(C(N2CCC(C)(NCCN(C)C)CC2)=O)=O)ccccc1[N+](=O)[O-] C12(C(=O)NC3C(C)CCN(c4c(C)c(Cl)ncn4)C3)CCC(CC1)C(C)(C)O2 N1(C(c2cnc(C(C)=O)s2)=O)CCOC(CCNC(=O)CC2CC3CC3C2)C1 Cc1[nH]nc2c1CC(C(N1CC3CC(NC(=O)Cc4cscn4)C3C1)=O)CC2 CCCC(C)(CCC)C(=O)N1C2CCC1C(CNC(=O)C(c1ccn(C)n1)C)C2 Cc1ccnc(NCC(C)(C2CC2)NC(=O)Cc2sc(C3CCC3)nc2C)n1 CC1CN(C(c2c(Cl)nsc2Cl)=O)CCCN1C(c1ccc(C(N)=O)cc1)=O C1(CC=C)CCCCN1C(C1C=CC(NC(=O)C(c2ccc(C)o2)C)C1)=O Cc1cc(C(=O)NC2COCCC2NC(C2CCC(C)(C)CO2)=O)cc(C)c1N CCC(CC)(CN=c1c(C#N)c[nH]c2ccc(Cl)cc12)NCC c1(C(N(C2CN(C(C(CC=CC)CC)=O)CC2(C)C)C)=O)[nH]cc2c1CCCC2 c1(C(N2CC(C)(NC(C(CC)C(C)C)=O)C2)=O)cc2c(o1)CCCNC2=O C12(C(=O)NC(c3cn(C)nn3)C)CCC(CC1)N(C(C1CCOC1(C)C)=O)C2 CCCCCCNC(=S)NC1CCSC1 c1(C2C(C(=O)NCC(C)NC(=O)C(=Cc3c[nH]cn3)F)C2)ccc(Cl)nc1 Cc1ccc(C(=O)NCC(C)C(C)(C)CN(C)C)c(F)c1.N12CC3CC1(C3)C2=O c1(OC)cc(CC2CCCN2C(=O)NCCc2ccc(F)c(F)c2)cc(O)c1 C(CC(C)C(F)(F)F)NC(c1ncn(CCNC(C2C(C)=CCS2)=O)c1)=O C1(NC(c2ccc(C)cn2)=O)CCC2CN(C(c3cc(Cl)cnn3)=O)CC2C1 c1(C(=O)NCCCN(C(=O)Cc2ccccn2)CC)cnn2c(C)ccnc12 N1(C(C(COCC)C)=O)CC2(CC(NC(c3cnc(O)cc3C)=O)CO2)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(F)CN3C)=O)C2)C)c[nH]c2ccc(F)cc12 C(=O)(C1=Cc2ccccc2OC=C1)NC1(CNC(C2C(C=C)CC2)=O)CCCC1 Cc1ccn2c(C(N3CCC(O)(CNC(=O)C#CC(=O)N(C)C)C3)=O)cnc2c1 C1(CNC(C2C(C(=O)OC)CCO2)=O)CCN(C(C2COC(=O)N2)=O)C12CC2 C1(C(=O)NC23C(NC(CCC#CC)=O)CC(CC2)C3)CCn2nnnc2C1 C#CC(CC(C)(C)C)NC(=O)CC1(C)CCN1C(=O)CN(C=O)CC N1(C(CCOC)=O)CCCC(N(C(=O)CCCc2sccc2C)C)C1 c1(N2CCC(COC)CC2)ccncc1S(=O)(=O)NCC1(C)COCCO1 N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c(C)[nH]c4ccccc34)=O)CC12 c1(NCC2C(NC(C(CC)OC)=O)CCCC2)cc2nncn2c(C)n1 Cc1nc(C(=O)Nc2cncc(C(=O)NC3CC34CNC4)c2)c(=O)[nH]c1C Cc1cc(C(=O)N(CCCOCCNC(C2C3CNC(=O)C23)=O)C)n(C)n1 CCCC(CCC)C(=O)N1CCC(NC(c2c(F)ccnc2Cl)=O)CC(O)C1 C1(CNC(COCCOCCOC)=O)C(O)C(O)CN1C(=O)CCS(C)(=O)=O N1(C(CC2N(C)CCC2)=O)CC2CC2(CNC(c2cnc(O)o2)=O)C1 C=C(C)C1OCCC1C(=O)NC1C2CC1N(C(c1cnncc1C)=O)C2 C1(NC(C2C(C)OCC2)=O)CCN(C(C2CNC(=O)C2)=O)CC1(C)C C(=O)(CC(C(F)F)N1CCOCC1)N.CC1CCC2(CC2)C1 C1(C(=O)NCC2CCN(C(=O)CN3CCCCC3)C2)CC(c2ccncc2)=NO1 C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(=O)C#CC2CC2)CCN1C N1(C(C(C)Cc2ccccc2)=O)CC(NC(=O)CC(C)C(F)F)CC(C)(C)C1 C1(C2CCCC2)(NC(C2C=CC(NC(=O)CC3CCC=CCC3)C2)=O)CC1 c1(NC(CC)C(N2CCCC(CCCC#N)C2)=O)ncnc2c1ncn2C1CC1 C=CC1CCCN1C(=O)C(C)(CO)NC(C1COCC1C(N)=O)=O C(=O)(C(O)C(F)(F)F)N(C)CCN(C(=O)CCc1cc[nH]n1)C c1(OC)cccc(C(=O)NC2CCN(C(=O)C(C)c3ccsc3)C2C)c1F CC1CN(C(C2OCCC2NC(=O)CC2CC(F)C2)=O)CCC1(F)F C1(C(C)NC(C=CCC)=O)CCN(C(=O)CC(=O)NCC)CC1 N1(C(C(C)OCC)=O)CC(C)(CNC(C2CC2c2ccncc2F)=O)CC1(C)C c1(C(=O)NC2CC(NC(C3(CC#C)CCCO3)=O)C2)sc(C(C)(C)C)nc1C C(=O)(C1=NOC(CNC(c2ccc(C(N)=O)[nH]2)=O)C1)N(CCOCC)C N1(C(C2(C(=O)OCC)CC2)=O)CC(C)C(NC(c2c[nH]cc2C2CC2)=O)C(C)C1 C1(CC=CC)CCCN(C(c2ccc(Br)cn2)C(=O)NCCCC2CC2)C1 CCC(CNS(C)(=O)=O)N=c1[nH]c(=NCC(CC)C2CCC2)[nH]c2cc[nH]c12 N1(C(COCC(C)C)=O)CCCC1(C)CNC(C1CN(S(C)(=O)=O)C1)=O N1(C(=O)OC(C)(C)C)CCCCC12CCCN(C(C1CC1(C)C)=O)C2 N1(C(c2ccn(CCOC)c2C)=O)CC2CCN(C(=O)C(C#N)C(C)(C)C)CC12 C(=O)(CC(C)(F)F)NCC(CC)NC(c1ncccc1-c1ccccn1)=O c1(CCC(N2CC(N(C(c3ccc(C(C)=O)o3)=O)C)C2)=O)ccc2[nH]ccc2c1 O=C(CCCCCc1ccccc1)NCC1CN(C(=O)C2=CCOC2)CC1O c1(OC)cc(C(=O)NCC#CCNC(=O)COCC(C)C)c(Cl)cn1 C(=O)(C1=CCC2CCC1N2C(C1(C)CC2CCC1C2)=O)NCc1cc(OC)no1 c1(OCC(=O)NCCC2CC(C(=O)N(CC(F)F)CCO)C2)cccnc1 CCCCCCCCCC(O)C(=O)N1CCCC(Cc2nccs2)C1 C1(CNC(c2cc(CCC)ncc2)=O)C(C)CCCN1C(c1cc(Cl)ccn1)=O C(=O)(C(C)CCC(C)(C)C)N1CCC(O)(CN(C(c2c(C)nc[nH]2)=O)C)C1 c1(COCC)cncc(C(=O)NC2(C)CC2)c1.c1(C(=O)N)ccc(C(F)(F)F)nc1 N1(C(CC(=O)NC)=O)CCC2(CCCN(C(c3cc(C#N)ccc3C)=O)C2)C1 N1(C(c2cnc(Br)s2)C(=O)CCCSC)CCC(c2ccccc2)CC1C c1(C(=O)NCCC(CC)NC(c2cocc2C)=O)c(C)nn(CC(C)C)c1Cl Nc1c(C(=O)NCCNC(c2[nH]nnc2-c2ccccc2)=O)cccc1F C1(C(C(C)NC(=O)CN(C)C(C)=O)OC)CCCCC1 c1(C(N(C2CN(C(=O)C(C)(C)C3CCCO3)C2)C)=O)ccc([N+](=O)[O-])cc1O C1(C(N(C2CCN(C(c3c(C(C)C)onc3)=O)C2)C)=O)C(C(F)(F)F)C1[N+](=O)[O-] c1(CC)cc(-c2cccc(CN(C(C)C)Cc3ccc(Br)cc3)c2)cc(N)c1 C(=O)(C(F)C1=CCCCC1)NCC1OCCCN(C(C2(C)CC2(Cl)Cl)=O)C1 C1(NC(C2CC(C)(C)O2)=O)CCN(C(=O)CCCCN2CCCCC2)CC1O C1(CNC(C2N(CCC)CCC2)=O)CN(C(=O)CCC#N)CCC1C N1(C(c2n(CCOC)ncc2)=O)CCN(C(C2CCC(C)(CC)O2)=O)CCC1C c1(C(=O)NCC2(NC(CC3C(C)(C)C(O)C3)=O)CCCC2)cc2n(n1)CC1(CC1)C2 c1(NCc2c(C)n(C)nc2C(=O)O)nn(C)c2ccccc12 N1(C(C(CSC)C)=O)CCCC2(C1)CN(C(=O)C(F)(F)C(F)(F)C(F)F)CCO2 C#CCC(C)(C(=O)Nc1cc(C)cnc1O)NC(=O)CC1CCC(C)(C)O1 N1(C(c2n(C)ccn2)=O)CC2CCC1C1CN(C(=O)CCc3ccnn3C)CC21 c1(C(N2CC(CNC(=O)C3CC3)OCC2)=O)cc(Br)c(F)cc1F C1(C(=O)N(CC(c2ccccc2)OC)C)(COC)CC=CC1.C1C(=O)N1 c1(NC(c2c[nH]nc2C2CC2)=O)ccc(CNC(=O)COCC(F)(F)F)cn1 C(CCCCC(=O)NCC(C)(O)CNC(=O)C(c1ccc(F)cc1C)O)OC NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2C(NC(C34CCC(C3)C4)=O)C2(F)F)c1 n1(C(C)C(=O)N(C2CCCS2)C)cc(C(C)(C)CC2CC2)nn1 N1(C(C2C(C)C(=O)C2)=O)CCOC(CN(C(=O)CCc2cn(C)cn2)C)C1 N1(CC(c2ccccc2)OC(C)C)CCC2C(CCCC2(F)F)C1 N1(C(C(C)NC(=O)CCc2nc[nH]n2)=O)CCC1(C)C c1(CC(=O)NC2CCCC(C(F)(F)F)C2)nsc2ccccc12 c1(C(N2C(C(=O)Nc3ccc(N(C)CC)cc3)CCCC2)=O)ncnc(O)c1F C(CC(C(=O)NC(C)C(O)C(F)F)NC(=O)C(O)Cn1cncn1)OCC c1(C(=O)NC2C(NC(=O)Cc3nc(C4CC4)cs3)CC2)snc(O)c1Cl c1(C(=O)NC2CCN(C(C(C)OCCCC)=O)C2(C)C)ccc2c(c1)B(O)OC2 c1(C(=O)NC2C(OC)CCC2)c(OC)cnnc1OCc1ccccc1 N1(C(c2csc(Br)c2)C(=O)NC)CC(SC)CC12CCOCC2 CC1(C)CCN(CCNC(c2ccc(CNC(C3CC=CCC3)=O)o2)=O)C1 c1(C(C)=O)ncc(C(=O)NCC2CC2CC(N2CCC(F)C2)=O)s1 C1(c2nc(C(Cc3ccoc3)OC)on2)(c2cccs2)CCCCC1 c1(OC)ccc(C(=O)NC2CC3CC2N(C(=O)C(C)(C)C#N)C3)cc1C(F)F CCCCCCCCC(=O)N1CCOCC1CCNC(=O)C(C)(CC)CO CC1(C)CCCC1CCNC(c1cccc(C(F)F)n1)=O C=CCCCC(C(=O)NCC(=O)NC(N)=O)NC(=O)CP(C)(C)=O c1(C(NNC(=O)c2ccccc2I)=O)cc(F)c(F)c(F)c1 C(CSC)(C(=O)NC(CC1CCCC1)C(=O)NC(C1(O)CCC1)C)OC c1(C(=O)NC(C2CN(C(=O)C3=CSCCO3)C2)C)ccnc2ccccc12 C#CC12CC1CN(C(=O)C(C)Cc1ccc(Cl)cc1F)C2 C1(CNC(C2(OC)CCCC2)=O)CCOCCC(=O)N1.CCOCC C1(C(=O)NC2CC3CN(C(CC4N(C)CCC4)=O)CC32)CCCC2(C1)CC2(F)F CC(C)S(=O)(=O)c1ccccc1C(NC1CCc2cccc(O)c21)=O N1(C(c2cccc(N)n2)=O)CCC2(NC(c3ccn4ccnc4n3)=O)CCCC12 c1(CC(=O)NC2CCN(C(C3CC(C)N(C)C3)=O)CC2)c[nH]c2ccncc12 c12cccc(c1)NC(=O)C2C.C1(C(N(C2CCC2)C(=O)OC)C)CCC1 N1(C(c2cc(C)ncc2C)=O)CCCC2(CCC2NC(c2cnccc2C)=O)C1 C12(NC(=O)CN3CC=CC3)CCOCC1CN(C(c1cccc(C(F)F)c1)=O)C2 c1(OC)ccc(CNC(C2C3CC2N(C(c2cncc(O)c2)=O)C3)=O)cc1 CC(C(=O)NCCC1CN(C(c2cc(Cl)c(Br)cn2)=O)C1)C(C)(C)C CCC(C)C(C(=O)NC1CC(NC(c2coc(-c3ccccc3)c2)=O)C1)OC c1(C(=O)NC2C(NC(c3cn(CCC=C)nn3)=O)COC2)cncn(C)c1=O N1(C(c2cc(CC)no2)=O)CCCC(C)(C)C1C(N1CC(Cc2ccco2)C1)=O C1(CNC(C=CC)=O)CN(C(c2c(-c3ccncc3)noc2C)=O)C(C)(C)C1 C(=O)(C1=NOC(C)C1)N(C(c1ccc(C(N(CCOC)CC)=O)cc1)C)C1CC1 C1(C(N2C(C)CC(NC(Cc3c(C)con3)=O)C2)=O)CCc2nncn2C1 C1(NC(C(C(C)C)OC)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1F Cn1cnc(CC(=O)NCC(C2CCOC2)NC(=O)COC2CCC2)c1 c1(C(N2CC(CC(C)NC(C(C(CC)C)O)=O)C2)=O)ccc(F)c(S(N)(=O)=O)c1 c1(CC)ccccc1C(CNC(C1(C)CC1)=O)NC(=O)CCCC1CCC1 CC(C)CCC(=O)NCC(=O)NC1C=CCN(C(=O)COCC2CCOC2=O)C1 n1(CC)c(CNC(=O)CN(C(=O)CC2CCOCC2)C2CC2)nnc1O C(=O)(C(CC(C)C)OC)NC1CC(NC(c2c(C)nc(CC)s2)=O)C1 c1(OC)ccc(CO)cc1C(=O)NC1CCC(N(C)C(c2cc(=O)cc[nH]2)=O)C1 c1(C(=O)NC2(CCOC)CCN(c3nnc(C(N)=O)s3)C2)ccc(S(C)(=O)=O)s1 C1(CC(=O)NCC(=CC(=O)NOCC2(CO)CCC2)C)CCN(C)CC1 C(C)(C(C)(C)NC(N(C)CCOC(C)(C)C)=O)NC(C(C)C1CCC1)=O c1(NCCCN(C(=O)C(C)OC)CC)ccc(C(=O)OC)cc1[N+](=O)[O-] C1(CCNC(c2cc(C(F)(F)F)no2)=O)CCCN(C(=O)CC2CCOC2=O)C1 CC1CCCCC1(CNC(=O)CN1CCCC1=O)NC(=O)CCCCO c1(-c2cn(CC3CN(C(c4occ(C)c4C)=O)C3)nn2)ccc2nccn2c1 c1(C(=O)NCC=CC(=O)NC2(C(C)O)CC2)cnco1 C1(C(=O)NCC2(O)CC(NC(c3ccc(=O)oc3)=O)C2)CC2CCC1O2 C(C)(C(=O)Nc1nc(-c2ccc(C)nc2C(F)(F)F)no1)(C(C)C)OC C#CCC(C)(C)C(=O)NCC(CC)N(C(=O)CCCNS(C)(=O)=O)C C1(CCC)CN(C(=O)COCCCOC)CC1NC(c1cc(C(C)C)on1)=O CC1(C)CCC(O)(C(=O)NCC2CC(O)(CNC(=O)CCc3cnco3)C2)CC1 c1(C(=O)NC(C(C)NC(C2CCC2)=O)C)ccncc1C(F)(F)F CC(COC(C)(C)C)C(=O)N1CC(OCCCCO)C1.C12CC1CC(=O)N2 c1(C(C)=O)cc(C(=O)N(CC(C)NC(=O)C(c2ccc(Cl)cc2)=O)C)c(C)s1 C1(NC(C2(CNC(C3(NC(C)=O)CC3)=O)CCCC2)=O)CC(C)(C)C12CC2 C(CC(=O)NCCC(C)OC)(C(F)F)NC(C1(CC)CC(C)(C)C1)=O C1(CN(C(C2(NC(Cc3c(C)con3)=O)CCC2)=O)CCC(C)C)CCC(C)CC1 c1(N2CC(OCCNC(C(N3C(=O)CCC3=O)CC)=O)C2)nccc(C)c1[N+](=O)[O-] c1(NC(=O)C=C2CN(C(=O)CCc3ccc(Br)c(F)c3)C2)ncc(Cl)cc1Br c1(C(=O)NCC2CCN(C(=O)Cc3ccc(Cl)cc3F)C2)ccc(Cl)c(Br)c1 c1(C(=O)NCC(CNC(C2(C)CCN(C)C2)=O)(C)O)cc(F)c2ccccc2c1 c1(OC)ccc(O)cc1C(=O)NC1CC(NCc2cc(Cl)ccc2F)C1 C1(NC(COC)=O)CCN(C(c2cc(Br)sc2Cl)=O)C(C)C1 O=C(C1=CC2CCCC12)N1CCN(C(c2ccc(-n3ccnc3)c(Cl)c2)=O)CC1 C(=O)(CCCCCS(N)(=O)=O)NCC1CN(C(c2ccc(OCC)nc2)=O)C(C)C1 c1(C(=O)NCC2CC3N(C(C(C)CO)=O)C(CC3)C2)ccc(Cl)cc1[N+](=O)[O-] C(C(C)(C)CC(C)O)NC(C1CN(C(C2(CC=C)CCCC2)=O)CC1F)=O N1(C(c2cnn(C(C)CC)c2)C(=O)NCC)Cc2ccccc2C1CCO CCCCC(CC)CC(=O)N1CCC(C)CC1C(=O)NCCN(CCO)CC N1(C(C2C(C)OC(C)C2C)=O)CCC(NC(=O)CCCCCO)C2(CCC2)C1 C1(CC)COCCN(C(C2CCCC(CNC(=O)CCC3(C)CC3)C2)=O)C1 N1(C(C(CC)SC)=O)CCCC1(CNC(=O)C(C)(C)c1cccnc1)COC C12(CNC(=O)CC3=CCCC3)CCCCC1N(C(=O)COc1ccccc1)CC2 N1(C(C2CN(C(C)=O)C2)=O)CCC(O)C(NC(c2c[nH]nc2C(F)F)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CC(CNC(c2cnc(SC)s2)=O)CC1(C)C N1(C(C2CCC3(CC3)C2)=O)CCCCC2(C1)CN(C(C1CCCCO1)=O)C2 C1(NC(=O)C(F)=CC2CC2)CS(=O)(=O)C2CN(C(=O)Cc3cscn3)CC12 Cc1cc(C(N2CCC(C(C)NC(=O)COCCCF)CC2)=O)c(C)nc1C c1(CNCC(C)C2CCC2)ccccc1CN(S(C)(=O)=O)C CCC(C)C(C(=O)NC1CN(C(C)C)CC1C)N(C(=O)C=C(C)COC)C c1(CC(N2CCC(N(C(C(CC)C)=O)C)CC2)=O)ccc(Cl)c(F)c1 C(=O)(CCCCC(F)F)N1CC(NC(=O)Cc2cnc[nH]2)C2C1C2 C1(CN(C(=O)COCP(C)(C)=O)C)CCCN(C(C2CC(N(C)C)C2)=O)C1 C1(NC(C(C2CCN(C(=O)CCC3CCC3)CC2)C)=O)CC2(CCCC2)C1 C(=O)(CCC(=O)NN(C)C)NC(CC)(CNC(C1C(C(F)F)C1(C)C)=O)CC C1(NC(C(C)CF)=O)COC2(C1)CN(c1ncnc3[nH]cnc13)C2 C12(C(=O)NCC(C)CNC(c3cc(F)cnc3O)=O)CCCC1CC(=O)CC2 c1(CC(N2CCOCC(NC(CCC(=O)N(C)C)=O)C2)=O)nnc2n1CCCC2 C1(CC(=O)OC)CCCCN1C(c1ncccc1OC)C(=O)NC1(C)CC1 C(C(N)=O)(C(F)(F)F)N(C(CCC)C(=O)O)C1CC1 Cc1n[nH]c(C)c1C(C)C(=O)N(CC(C)N(C)C(c1ncccc1CO)=O)C C1(C(=O)OC)C(F)(F)C12CC(NC(=O)NC(Cc1ccc(C)cc1)C(C)(C)C)C2 N1(C(c2cccc(N(C)C)c2)=O)CC2CC1CC2NC(c1cc(O)ncc1F)=O C12C(CC(CC)C1)C(=O)OC(=O)N2C1CC12CN(C(=O)OC(C)(C)C)C2.CC.OC C=C1CCC(C(N2CC3CC3(CNC(=O)C(C)Nc3nc(C)cs3)C2)=O)CC1 C1(C(=O)OC)COCCN(C(=O)C(=O)N(C2CC(C(F)F)C2)C)C1 c1(NC(C2OCCN(C(CSCC)=O)C2)=O)c(F)c(F)c(Cl)c(F)c1F C12(CCC1)C(=O)N2C.C1(COC)CCN1C(=O)CN(C(=O)C(C)C)C C(=O)(C(=O)NOC)NC(c1ccccc1)C(=O)NC1(C=C)CCC1 c1(C(=O)NCC(C2CCN(C(=O)CN3CSCC3=O)CC2)(C)O)ccncc1Cl N1(C(COC)=O)CCC(OCCNC(c2cn(-c3cccnc3)nn2)=O)C1 C1(NC(C2(C#N)CC2)=O)COC2(CCCN(C(c3cc4ncccc4[nH]3)=O)C2)C1 CCCC(C(=O)OC)C(=O)N1CCOCC(NC(C2CC(C)(C)CCO2)=O)C1 c1(C(N(C)CC2COCCN2C(C2CSCCS2)=O)=O)cnn2c(=O)cc[nH]c12 c1(CC(C)C)cc(C(=O)NC2CC3CC2N(C(=O)C(C)(F)F)C3)cc(O)n1 CC1(C)CC(C)(NC(c2ccc3[nH]ccc3n2)=O)CN1C(=O)CNS(N)(=O)=O Cc1cccc(-c2cn(C3CCN(C(C4CCCCS4)=O)C3)nn2)c1F C(C(C#Cc1cccnc1)OCCO)NC(c1cccc(C2CC(=O)NC2)c1)=O C(=O)(C(C)CC(C)(C)C)NCCC1(O)CCN(C(c2cnc(C)[nH]2)=O)C1 O(NC(=O)CCC(C)N(C)C(C1(CF)CCOCC1)=O)Cc1cccc(C)n1 c1(C(=O)NC(C)CCNC(=O)CN2CCOC2=O)cc(O)cnc1Cl Cc1c(CCNC(=O)CN(C(=O)C=C=C(C)C)C)cnn1C c1(SC)cc(C)c(C(=O)NCC2CN(C(=O)CCc3cncc(O)c3)CCO2)o1 c1(C(N2C(CC(=O)Nc3c(OCC)cccc3)CC2)=O)ncc(F)cc1N Cc1nsc2ncc(C(N3CCCCCC3CNC(=O)CN(C)C(C)C)=O)cc12 c1(CC(C)NC(=O)CC2CCCN2C(c2cnc(C3CC3)o2)=O)cccnc1 O=C(NNc1ccc(N2CCOCC2)cc1)c1ccc(CO)cn1 N1(C(CS(C)(=O)=O)=O)CCCC2(C1)CN(C(c1ccc(C(F)F)cc1)=O)CCO2 C(=O)(C(C)CCC(C)(C)C)N(CCCNC(C(CC(C)C)O)=O)CCO c1(C(N2CC(CC#C)OCC2)=O)cc(O)nc2c1CN(C(=O)CC(C)C=C)CC2 CC(N=c1cc2ccccn2[nH]1)C(C)n1ccnc1 CC(C)CCCC(=O)NC(CCN(C(=O)CC1CC1(C)C)C)C(C)C N1(C(=O)COC(F)F)CCN(C(c2ccc(CO)nc2)=O)C(C2CC2)C1 N1(C(C2CCCC(=O)N2)=O)CC(NC(=O)C=Cc2cncnc2O)CC2(CC2)C1 c1(C(=O)NCC(CC(C)C)NC(C2CNC(=O)N2C)=O)c(O)cccc1Cl C(C(=O)N=c1cc(C)o[nH]1)N1CCC(CCCNC(CCCC=C)=O)CC1 c1(C(N(C)CC2N(C(C(N3CCCC(O)C3)C)=O)CCC2)=O)nc(Cl)c(Cl)s1 c1(OC)cc(C(=O)NC2CCN(C(=O)C(C)(C)C)CC2CO)c(Cl)cc1Cl c1(CC)sc(=N)[nH]c1C(=O)NCCOCCN(C)C(C1(C)CCCO1)=O N1(C(C(C(CC)CC)O)=O)CC(NC(c2cccc(C)c2)=O)CC12CCOCC2 C1(CNC(C(C)OCC2CC2)=O)(COC)CCN(C(S(=O)(=O)C2CC2)=O)CC1 c1(C(N2CCC(NC(c3c(C)nn(C)c3)=O)C2)=O)ccc(=O)n(C(C)C)c1 c1(C(N2C(C)C(O)CC2)=O)cc(O)nc2c1CN(C(C1CCN(C)C1C)=O)CC2 Cc1ncnc(C)c1C(=O)NC(C)CCCCNC(c1cnc(N(C)C)nc1)=O N1(CCC)CCCC1C(N1CCC(C(=O)NC(c2cccs2)C)C1)=O C1(NC(Cc2c(C)n(C)nc2)=O)CC2(C1)CC(CO)C2.C12CCN(C1C)C2=O C1(C(=O)Nc2cccc(COC)c2)N(C(=O)CCc2cccs2)CCC1(C)C C1(CNC(C(C)NS(C)(=O)=O)=O)CN(C(c2ccc(F)cn2)=O)CC(C)(C)O1 CC1(C)CN(CCC2CCN(CC(F)(F)F)CC2)C1C1CCCO1 CCCCCC(O)CC(=O)NCc1ocnc1C(N1CCCC1(C)COC)=O C1(C(N(C(C)C)CC2CCCO2)=O)CC2C=CC1C2.c12ccc(s1)CNC2=O CC1(NC(c2cccc(Oc3ccc(F)cc3)c2)=O)CCCN(C(=O)CO)C1 N1(C(C=CC(C)C)=O)CCOCC(NC(c2cccc(SCC#N)c2)=O)C1 Cc1ccc(C(=O)NCc2cn(C3CCN(C(c4cnsn4)=O)C3)nn2)c(Cl)c1 CCCCCC(C)CC(=O)N(CCC(=O)Nc1cccc(CC)c1)C CC1CCC(C)(CNC(=O)C(=O)NCCNC(c2cccc(O)n2)=O)C1(C)C Cc1c(C(N2CCN(C(=O)CC(C)C)CC2CC(F)(F)F)=O)sc2ccccc12 N1(C(c2cnn(C)c2Cl)=O)CCC2(CCN(C(C3CC(CCO)C3)=O)C2)C1 CC(F)(F)CCC(=O)N1CCC(N2CCN(C(c3ccnc(F)c3)=O)CC2)CC1 c1(C(N2CCC(NC(C(C)C3CC3)=O)C2)=O)ccc2c(c1)OCCO2 C1(O)(CN(C)C(C2CC(=O)CN2C(C2(C)CCCO2)=O)=O)CCCCC1 C(=O)(C1COc2ccc(Cl)cc21)NC12CC3CCC(C1C2)N3C(C(=O)N(C)C)=O O=C1CCN2C(=O)C2N1.C(CS(=O)(=O)O)SCCCOC1CCCC1 C1(C(=O)NC(CNC(c2c(Cl)ccc(C)c2)=O)C(C)C)Cc2n[nH]cc2C(=O)N1 C(CN=c1cccn[nH]1)NC1CC1C1CC1.O=C1NCCN1 N1(C(c2c(C)nc(C(C)C)cc2)=O)C2CCCC1CN(C(C1COCCO1)=O)C2 c1(N(C2(C(=O)O)CCC2)C)ncnc2c1SCCC2 Cc1ocnc1C(=O)NC(C(=O)NCc1cn(C)cn1)C1CCC1 N1(C(CCCC)=O)C2CCC1C(F)C(NC(C1CCSC1)=O)C2 C1(C(N(CC(O)CNC(=O)CCc2ccon2)C)=O)CC(C)(C)SC(C)(C)C1 c1(N(C)CC2CCN(C(=O)COc3ccsn3)C2)ncc(S(C)(=O)=O)cc1Cl CS(=O)c1ccc(CC(=O)NC2CN(C(c3ccc(O)nc3)=O)CC2O)cc1 n1(CC(=O)NC2CC2Cl)cc(CN(CC)CC2CCCCO2)nn1 c1(CN2C(CNC(C3C(C)CCC3)=O)CC2)ccc(N2CCCC2)cc1 c1(C(=O)NCC2C(NC(C(CC)OC)=O)CC2)ccc2c(c1)nnn2C N1(C(C2(C#C)CCC2)=O)CC(NC(=O)CCc2cc(C)cc(C)c2)C2(CC2)C1 c1(C(CC(=O)OC(C)(C)C)N)ccc(OC(F)(F)F)cc1.C1(=O)CCCCO1 C1(C(=O)NCC2CCN(C(c3ccoc3)=O)C2)C2CCC3(COC(=O)C13)O2 N1(C(C2CC(C(C)C)C2)=O)CCCC1c1cn(C2(C(=O)O)CC2)nn1 N1(C(CNS(CC)(=O)=O)=O)CC2CC1CN(C(C1CCC(C(C)C)CC1)=O)C2 N1(C(c2nc(Cc3cc(F)ccc3F)no2)C(=O)NC)CCCC(F)(F)C1 C(=O)(C(CCC)OC)N1CCC(C(C(=O)NC(C=C)(C)CC)(C)C)C1 C#Cc1cccc(C(=O)NCC2CN(C(c3ccnc(F)c3)=O)CCC2C)c1 N1(C(CCOCCNC(C(COCC)N=[N+]=[N-])=O)=O)CC=CC12CCOCC2 c1(C(N2CC(CNC(=O)COC3CCCC3)C2)=O)cc(F)sc1Br C(CCC(=O)NC1(CCN(C)C)CCOC1)=C(C)C.c12ccc(s1)C(=O)NC2 C(=O)(C#CC1CCCOC1)NCCN(C)C(C1(C)CCCNC1=O)=O C1(CC(=O)NCc2c(C(=O)NCc3onc(C)n3)cco2)CCCC(=O)N1 N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C(F)(F)CC1 C12(C(=O)NC(C34CCC(CO3)C4)C)COC(C1)C(NC(=O)C#CC1CCC1)C2 C1(NC(CCC2C(C)C2)=O)CN(C(c2cc(Br)cn2C)=O)CC12CCOCC2 c1(C(N2CCC(F)(CNC(C3C(C)(C)C3)=O)C2)=O)ccc2c(c1)CC(C)(C)C2 c1(C(=O)NCC2C(NC(C(C)N(C)C)=O)C2)c2n(c(=O)n1C)CCCC2 Cc1ccc(C)c(C(=O)NCC(C2CC2)NC(c2cc(C(F)F)c(C)s2)=O)c1N N1(C(c2cn(C)nc2O)=O)CC(NC(C2C=CCS2)=O)CC2(CCC2)C1 c1(CC)cc(C(=O)NCCCN(CCO)C(c2cnsc2)=O)ccc1C C1(NC(c2cc(Br)no2)=O)COC2CN(C(c3ccnnc3)=O)CC12 C(=O)(CCC(C)N(C)C)NC(C1N(C(C(=O)NCC)=O)CCC1)C N1(C(C#CCC#N)=O)CC2CCCN(C(c3ccc(Br)cc3Cl)=O)C2C1 C1(O)(CNC(C2C(C)(COC)C2)=O)CCN(C(c2cnc(C3CC3)s2)=O)CC1 c1(C(N2C(C)(CNC(c3cc(CF)on3)=O)CCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nn(-c2ccccc2)cc1C(N1CCCC1C(C)NC(=O)C=C(Cl)Cl)=O C1(C(=O)NC2C=CC(C(N(C(C3CCC3)C)CC)=O)C2)CC12CCOCC2 C(=O)(CCCCC(C)(C)C)N1CC2C(N(C)Cc3nc(CC)sc3)(CCC2)C1 N1(C(c2c(CSC)cccn2)=O)CC2CCN(C(C3CC(SC)C3)=O)CC2C1 c1(OC)ccc(CC(=O)NCC2C=CCN2C(c2cccc(Cl)c2Cl)=O)cc1F C(=O)(C(C)(C)c1cncnc1)OCCN(C=O)C(c1ccccn1)=O CC1COC(C)(C)CN1C(c1cc(O)nc2c1CCC2)=O N1(C(CCC(CC)C)=O)CCC(C2CCN(C(c3cncc(Br)c3)=O)C2)C1 N1(C(COCCCCCC)=O)CCCCC1C(C)(C)CNC(=O)Cc1cnoc1 C(c1cncc(-c2nn[nH]n2)c1)=CC1CCC(C)N1C(c1ccccc1Cl)=O C1(C(N(CC=C)OC)=O)CCC2CCC1N2C(=O)Cn1cc(Cl)cn1 c1(C(N2CCC(CN(C(=O)Cn3cccn3)C)CC2)=O)cc([N+](=O)[O-])cnc1O CCC(F)C(=O)N1CCC(N(C(=O)CCC=CCC=C)CCO)C1 C1(C(=O)NCC(CC)NC(=O)OC(C)(C)C)CCC(CC)CC1 c1(NC(C(C(CC)O)C)=O)ccc2nccn2c1.C12(COC)C=CCN1C2=O Cc1oc(C(=O)NCCOCC(F)(F)F)cc1CO.N12CCC1C2 C(=O)(C(Cc1ccco1)CC)NC(c1c(C(N(CC(CCC)O)C)=O)con1)C N1(C(CC2CC(NC(=O)CNc3ncccn3)C2)=O)C2COCC1C2 c1(C(N2CC3(CC(NC(=O)CC4CS(=O)(=O)C4)C3)C2)=O)noc2cc(Cl)ccc12 c1(NC2C(NC(c3c(O)ccc(F)c3F)=O)CCC2)nc2ccccc2s1 N1(C(CC(CC(C)C)NC(CC2C(CC)C2)=O)=O)CCC12CCC(C)CC2 c1(COC(=O)NC2CCCC2n2cccn2)cccc(F)c1 c1(C(=O)NC(c2cn(-c3c(C)ccnc3)nn2)(C)C)ccc(S(N)(=O)=O)c(C)c1 CC1(C)CCCC(C(=O)NC(CNC(c2cnc(=N)[nH]c2)=O)C2CC2)O1 c1(OC)ccc(F)c(C(N2CCCC2C(C)NC(c2cncn2C2CC2)=O)=O)c1 C(CC(=O)NOCC1CCCO1)NC(C1CN(C(CC2(NC(C)=O)CC2)=O)C1)=O Cc1cc(F)c(C(=O)NC(C2CCOC2)CNC(=O)CC(C)(C)C)cc1F C1(OC)CC(NC(=O)Cc2ccc(C(=O)CN(C)C)cc2)C1(C)C C#CC1(NC(C2CCC(CNC(=O)C=CCN3CCC3)C2)=O)CC(F)(F)C1 C1(NC(=O)COCC2CCCC2)CCC2(CCCN2C(c2nncs2)=O)CC1 c1(C(=O)N(CCC(N2CCC(F)(CF)CC2)=O)C2CC2)c[nH]c2ccccc12 CC(C)CC(O)C(=O)N1CCN(CCCNC(c2cc(Cl)no2)=O)CC1 n1(CC#C)c(C(N2CCOCC2CC(C2CC(F)(F)C2)=O)=O)cc2ccccc12 c1(C(=O)NC(CNC(C2CCC(C)C2)=O)C)cc(S(C)(=O)=O)co1 C(=O)(C(O)CCCNC(C1(C#N)CC1)=O)NC(C)(C)C(N)=O c1(OC)ccc(C(=O)N(CCN(C(=O)C(C)N(C(N)=O)CC)CC)CC)cc1C N#Cc1ccncc1C(=O)NCC1OCCC1C(=O)N(CCCO)CCCO c1(OC)cncc(C=CC(=O)N(CCNC(c2ccc(F)c(Cl)c2)=O)C(C)C)c1 N1(C(C(C)n2ccnc2)=O)CCOC(C(=O)Nc2ccc(F)cc2)CC1 C(=O)(CCN(OC)C(=O)c1ccc(O)c(F)c1)NC1C(c2c(OC)cccc2)C1 N1(C(C(=O)N(CC)CC)=O)CCN(C(=O)C(F)n2cccn2)CC1CF C(=O)(C1=CCC(NC(c2cc[nH]c2)=O)C1)NCCC1C(C)CCO1 CC(C(=O)NNc1ccc(Br)c(F)c1F)C1CCCO1 N1(C(C2(C(=O)OC)CC2)=O)CCC2(CC(C(=O)N(C3(C#N)CC3)C)=NO2)C1 c1(CC)nc(-c2nc(-c3ccc(N(C)C)cc3)nn2-c2nc(Br)nn2C)sc1C CCCCCC(=O)N1CC(NC(c2csc(-c3cccc(C)n3)n2)=O)C(C)C1 c1(C(=O)NCCC(C(N2CCCC(C)(O)C2)=O)OC)ncc2ccccn12 c1(SC)ccc(CCCC(=O)NC2C3CC2N(C(=O)CC2CCC(C)C2)C3)cc1 C1(C(=O)NC(CNC(=O)C=C2CCCCC2)CO)(CC)CCC(F)(F)CC1 CC1(O)CCCN(C(c2c[nH]nc2CNC(=O)CC2CCC(=O)N2)=O)C1 c1(CNC(C)=O)cccc(C(=O)NCC2CC2CNC(c2ccncc2Cl)=O)c1 C(CC(C(C)(C)C)NC(c1cccc(CF)c1)=O)N(C)C(C1CSC1)=O CC(C)CC(C(=O)N1CC2CC2C2CC12)ONC(=O)CC1C=NN(C)C1=O c1(C(=O)NCC2(C(F)F)CCN(C(c3c(SC)csc3)=O)C2)c(C)cnnc1O c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc(CO)c(F)c1 C1(C)(NC(=O)NC(C)CC2(CO)CCC2)CC1(C)C c1(C(=O)NCC(C)NC(=O)Cc2ccccc2Br)cc(C#N)c(F)cc1F Cc1c(NC(c2nc(-c3ccccc3)oc2C(C)C)=O)cnn1CCO C1(C(N2CCC(O)(C(C)NC(CSC)=O)C2)=O)CCC(O)CN1C C(=O)(CCCC#Cc1ccccc1)NC(C)CNC(=O)CSc1ccc(O)cc1 c1(NCCNC(C)=O)ncc(-c2csc(NC(=O)N(C)C)n2)cn1 N12CCOC(C1)C2.c1(NC(=O)C(C2CCOCC2)F)csc(CN(C)C)c1 c1(OC)cc(OC)cc(CN2CCC(C)(C(=O)Nc3cc(F)cc(Br)c3)C2)c1 N1(C(CC2(OC)CC2)=O)CCC2CCN(C(c3cc(O)nc(O)c3)=O)CC2C1 CC(C)C(=O)CCCN1CCN(C2CCCCC2O)CC1 c1(CNCC(c2ccc(C3CC3)cc2)OCC)cc2n(n1)CCC2 C(=O)(C#CC1CCC1)N1CCC(C(C)NC(c2ccn(CC)n2)=O)C1 C(=O)(N=c1[nH]nc(CO)s1)NCC(CC)O c1(CN(c2ccccc2)C(=O)NC2CCCC(COC)C2)ccnc(C)c1Cl c1(C(=O)OC)cc2c(c(S(=O)(=O)Nc3cccc(N4CCCC4=O)c3)c1)CCC2 CCC(C)C(C(=O)N(C(C)(C(=O)NC1CC1CC(C)C)C1CC1)C)OC c1(N2C(C(N3CC4CCC(C3)O4)=O)CCC2)ncc(Br)cc1Br Cc1cncc(C(=O)NC(C2CCOC2)CNC(=O)CN(C)C2CC2)n1 C1(CCNC(CC2(C=C)CC2)=O)CC12CCN(C(=O)C(C)CC)CC2 C(=O)(CC1CCC(=O)c2ccccc21)Nc1c(OC)cccc1F c1(C(=O)NC2C=CCN(C(C(CC)CC)=O)C2)ccc2c(c1)CN(C)C2 N1(C(CC2C(OC)COCC2)=O)CC2CC(NC(c3ccc(F)cc3)=O)C1C2 C1(C)(C(C)C)CC1C(=O)N(CCNC(=O)Cc1cc[nH]c1)CCOCCO C1(CNC(CCN(CCC)C)=O)CN(C(c2cscc2F)=O)CC(C(F)(F)F)O1 N1(C(CN(C)C(N)=O)=O)CCCC(O)(CNC(C2(C)CCC(F)(F)CC2)=O)CC1 c1(C(c2ccccc2Cl)(C)NC(=O)C(=O)NC2CC3CCC2C3)ccccc1F C(=O)(CCC(C)(C)NC(c1cn(C)c(=O)n1C)=O)NCc1c(C)csc1 CCC(CC(F)(F)F)C(=O)N1CCC(CNC(c2cnc(C(=O)OC)cn2)=O)C1 C(Cc1ccccc1C)(N=c1cc(C)n2[nH]c(=N)nc2[nH]1)OCC Nc1cc([N+](=O)[O-])ccc1C(=O)NCC1CC1NC(c1ccccc1[N+](=O)[O-])=O N1(C(=O)CC2CC3CCC2C3)CC2CN(C(C3(Br)CC3)=O)CC(C1)O2 C#Cc1ccc(C(=O)NC(C)(C)C(N2CCC(O)(CO)C2)=O)cn1 C(=O)(C1CCCc2ncccc21)NC12C(CN(C(c3c(C)nn(C)c3Cl)=O)C1)C2 c1(C(N2CC(NC(C=CC(CC)=CC)=O)C(C)(C)C2)=O)ccc2nncn2c1 Cc1cccc(N2CC(C(=O)NC(C)Cc3ccccc3I)CC2=O)c1 C(C(N=[N+]=[N-])C(=O)N1CCCC1(C(=O)NOCC1(C)CC1)CC)OCC N1(C(c2cc(C)oc2)=O)CCC2CN(C(=O)C(c3csc(=N)[nH]3)=O)CC12 S(=O)(=O)(c1ccc2c(c1)CN(CCC(N)C(F)(F)F)C2)NC(C)(C)C Cc1nc(NCc2ccc(N(C)C)c(C)c2)cc(=NCC2CCOCC2)[nH]1 C12(CNC(C3CC(O)C3)=O)CCCOC1CCN(c1ncnc3cnccc13)C2 C(=O)(N=c1ncnc2[nH][nH]c(C)c1-2)C1C(NC(c2cc(C)cc(C)n2)=O)C1 N1(C(=O)CCc2cnccn2)CC2CCC2(CCNC(C2(F)CCCC2)=O)C1 C1(CNC(C2C(C(C)O)C2)=O)CCN(C(C2(C(C)C)CNC(=O)C2)=O)CC1C c1(C(=O)NC(C(=O)NCc2c(C)nc(C)s2)CCF)ccc(C)c(O)c1 n1(CCC)nc(C)cc1C(=O)NCC(C1CCCC1)NC(=O)CC1CSC1 c1(C(=O)NCC2CC(COC)CN2C(=O)CCCC2CCC2)cc(Cl)cc(Cl)n1 C1(C)(NCCCC(=O)OC(c2cscn2)C)CCN(Cc2ccccc2)CC1 c1(C(=O)NCC(CCCC)NC(=O)C(C)=C2CCC2)ccc(OC(C)C)cc1F c1(C(N(C(C)CNC(=O)CC2CCOC(C)(C)C2)C)=O)c[nH]c2cnccc12 C1(C(=O)NC2C(CC=C)CCC2)CC(O)CN1C(C1CN(C(N)=O)C1)=O C=CCCCCCC(=O)NC1CCN(C(=O)OCCC(C)C)CC1F c1(C(N2C(C)CC(c3ccccc3)C2)=O)cc2cccc(Br)c2cn1 c1(C(=O)NC2CCCC(C(=O)Nc3cnoc3)C2)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCC(C)(C)NC(C(C(COC)C)C)=O)cc(C)c(F)cc1F N1(C(COC(C)=O)=O)CCC2(NC(=O)Cc3ccc(F)cc3Cl)CCCCCC12 CCC(CC(=O)NCC1CC(NC(c2ccc(C(=O)OCC)nc2)=O)C1)C(C)C N12CCC(C)(C)C1C2=O.N1(C(C2CC(SCC)C2)=O)CCCC1Cn1ccnn1 N1(C(CC(CC)C(F)F)=O)CCC2(CCCCC2NC(=O)C=CCOC)CC1 n1(CC(=O)OC)cc(NC(C2CC(C(C)(C)C)C2)C)c(C)n1 C1(C(N2CC(CCNC(c3cc(C)oc3)=O)OCC2)=O)CN(S(N)(=O)=O)C1 c1(C(=O)NC(CN(C)C)C(=O)NCCN2CC=CC2)cccnc1S N1(C(CC(CC#C)c2ccccc2)=O)C2CCC1CN(C(C)=O)CC2 c1(CC)cc(F)c(S(=O)(=O)N2CC(C(=O)NC)CC2C(=O)OC)cc1F Cc1cc2c(cc1NC(=O)NCCOC(C)C)CCO2 N1(C(c2c(C)ccnn2)=O)CCCC(CO)(NC(c2cccs2)=O)C1 Cc1noc2ncc(C(N3CC(NC(C4(C)CC4)=O)C(O)C3)=O)cc12 C1(OC)CC(C(=O)NC(c2nc[nH]n2)CO)N(C(c2cscn2)=O)C1 C1(n2cc(-c3n(C(C)C)ncc3)nn2)CN(C(=O)CCP(C)(C)=O)CCC1O Cc1nnc(CCC(=O)N(C)CCN(C)C(c2cc(O)cs2)=O)n1C O=S(=O)(c1ccc(NCCN2CCOCC2)cc1Br)N1CCCC2(CCSC2)C1 c1(NC(C)CCC(F)(F)F)ccc(S(=O)(=O)NCC2(C)CCCOC2)cc1C#N N#CC1(C(N2CC(CCCCNC(C3CC34CCCCC4)=O)C2)=O)CCSCC1 c1(OC)ccc(C(=O)NCC2C3CN(C(C4(F)CC4)=O)CC23)c(OC(F)F)c1Cl C(=O)(C(Cc1ccccc1)CC(C)C)NC1CC(NC(C(CC)CC)=O)C1 C1(C(=O)NCc2cc(F)ccn2)CCC2(CC1)CCN(C(=O)C(F)(F)F)C2 N1(C(c2c(CC)con2)=O)CC(C2(NC(=O)COc3ccc(Cl)cc3F)CC2)C1 CCC(COC)C(=O)N1CCC(CC(=O)NC(C)CC(C)CC)CC1 Cc1cc(C(=O)NC2CCC2NC(c2csc(Cl)c2Cl)=O)ncn1 CC(C)C(CC(=O)N1CC2C(CO)C2C1)NC(=O)CC1CCOC1(C)C C1(CNC(CC2CC(C(C)=O)C2(C)C)=O)CC(C)CN(C(c2ccns2)=O)C1 CC1CCCCC1(CNC(=O)CCCCC1CCC1)NC(C1CN(C(C)C)C1)=O Cc1cc(O)nnc1C(=O)NCC1CN(C(C2CCC(C)CC2)=O)CC1C c1(C(=O)NCC2CN(CC3(c4ccccc4)CCCO3)C2)cccc(O)n1 N1(C(C2(NC(=O)OCC3(CO)CC=CC3)C(C)C2)=O)CCC12CCC(O)CC2 C1(C2CC2)(CNC(CN(CCOC)C)=O)CCN(C(C2(C3CCCO3)CC2)=O)C1 c1(OC)ccc(C(=O)NC(C)CCCNC(C2(C)CCOC(C)C2)=O)cc1C C(=O)(CCOCC(C)(C)C)N(C1(CC(=O)NC(c2ccns2)C)CC1)C C(=O)(C(C)CC(N)=O)NC1C(CNC(c2c(C(C)C)scn2)=O)CC1 C1(CNC(c2nc(C)sc2)=O)CN(C2CCN(C)C2=O)CCC1(C)C C1(c2n(C)ccn2)(C(O)NC2CCCC2C(C)(C)C)CCOCC1 c1(C(=O)NC(CNC(CC2CCC(C)C2)=O)(C)C2CCC2)ncc2ccccn12 C1(C(N(CCC#N)Cc2ccccc2F)=O)C2C=CC(C2)C1CN N1(Cc2cccc(C)c2)CCCC(NC(=O)CNC(=O)CC(C)(C)C)CC1 C1(NC(c2nnn(CC)c2C)=O)CC(NC(c2occc2F)=O)C12CCC2 N1(C(CC=CCNC(C2C(C)CCC2)=O)=O)CCCC2(C=CCO2)C1 c1(N(C(C#C)C)C)nnc(C(C)OC(C)C)n1CC(C)C C1(CC(=O)NCC2N(C(C3=CN3C)=O)C3C(C2)C3)CN2CCN1CC2 N1(CCC(c2nnnn2CCCF)C2CC2)CCc2ccccc2C1=O.C=C(C)CN c1(-n2c(C(=O)NC3CC(CNC(CCOCC#C)=O)C3)cnc2)ccccc1Cl C(=O)(C1CCCc2ccnn21)N1CCC(O)(CN(C)C(c2ccc(F)cn2)=O)C1 N1(C(C(CC=CC)CC)=O)CCC2CN(C(=O)C=Cc3sc(Cl)nc3Cl)CC12 c1(C(N2C(CNC(c3n(C(C)C)ncc3)=O)CCC2)=O)c(Br)cc(F)c(F)c1F CC(CC(=O)N1CCCC1(C)CC(=O)NC(C1CCC1)C1CC1)C(F)(F)F c1(OCCC)ccc(C(N2CCC(C)(CNC(=O)CCOCC(F)F)C2)=O)cc1 C(=O)(CCCCC#N)NCC1(F)CCC(CNC(C(C)Sc2ccccc2)=O)C1 C(=O)(CC(F)(F)C(C)(F)F)N1CCC2(CN(C(C(C=C)(C)CC)=O)C2)C1 C1(C(=O)OCC)C(C(=O)NCC2CN(C(C3CCN3C3CCCC3)=O)C2)C1(C)C Cc1cc(C)c(C(N2CC(C(F)(F)F)C(CNC(C3CCCC3)=O)C2)=O)c(=O)o1 Cc1cc(C)c(NC(=O)C(C2CC23CCCCC3)N2CCC(F)(CO)C2)c(C)c1 N1(Cc2onc(CCC)n2)CCC(NC(=O)CSc2ncc(C)o2)CC1 C1(CNC(=O)CCC2CCC2)C2CCCC1N(C(c1nnc(C3CC3)o1)=O)C2 C1(NC(CCC=C(C)C)=O)CC12CCN(C(c1nn(C)cc1Br)=O)CC2 CC1Oc2c(F)cccc2C1NC(c1ccc(C#N)cc1Br)=O C1(C(=O)N(C)CCC2CCC2)(SC)CN(C(C2CCCC2O)=O)C1 C1(NC(C2SCCS2)=O)CCN(C(C2CC2F)=O)CC1O C1(C(N2C(C3(NC(CN4CC(C)(OC)C4)=O)CC3)CCC2)=O)CC2(CCCC2)C1 CCC1=C(C(=O)NCCOCCCN(C)C(C23CC4CC2C3C4)=O)SCCO1 N1(C(C(CC)NC(C)=O)=O)CC2C(C(=O)NC(C)CC3CCCCC3)C2C1 C1(C(=O)NCCC2(O)CN(C(C3(C)C=CCCC3)=O)C2)Cc2nccn2C1 C1=CC2=CC(=NCN1CC1CCC1)NC(=NC1CC3CC3C1)N2 c1(C(N(C2CCC23CCNCC3)CCNS(CC)(=O)=O)=O)cc(F)ccc1[N+](=O)[O-] N1(C(c2c(CC)csc2)=O)CCCC12CCN(C(c1cscc1OC)=O)C2 C1(CCC)CN(C(c2c(C)cnn2C)=O)CCN1C(C1CC1c1ccccc1)=O C1(C(=O)NC2CN(C(c3ncn(C)n3)=O)CC2O)CCCCNC1=O C#CCC(C)(C)C(=O)NC(C)CCN(C(=O)C(C)Oc1cccc(C(C)=O)c1)C C(=O)(CCCCc1cnn[nH]1)N(C1CC(N2CCCC2)C1)C=O C1(CC(=O)OC)CCN(CCn2cccn2)CCC1(F)F C(=O)(C(C)CC(C)(C)C)N(C(C(=O)N(C)Cc1ncc(C)o1)(C)C1CC1)C c1(C(=O)NCC(C2CC2)NC(c2cccc(C(C)(C)C)c2)=O)cccn(O)c1=O c1(NC2CCN(C(COCCOCC)=O)CC2)nc(C)cc(C#N)n1 N12CCC13CN(C3)C(=O)C2.c1(CS(=O)(=O)N(C)C)cccc(F)c1 C1(C(N)=O)COCCN(CC(=O)NCc2nnc(-c3ccccc3F)s2)C1 C1(CN(C(=O)CCCCN2CCCCC2)C)CCCN(C(=O)COCCCF)C1 c12ccccc1OOC(=O)C2.C1(NCc2ccccc2)CC2CNC1C2 Cc1[nH]nc(C(=O)NC(C2CCN(C(c3ccc(N(C)C)cn3)=O)C2)(C)C)c1F C(=O)(C(C)(C)C(N)=O)N1C(C2(NC(C3CCN(CCC)C3)=O)CC2)CCC1 CN1CC(C)(C)CC1C(=O)N(C(c1ccccc1)CNC(C1CCC1)=O)C C1(N(C(CCOC)=O)C)CC2CC2C1.C12CC1C(=O)N(C1CC1)CC2 c1(C(=O)NCC2(C)CCN(C(=O)Cn3[nH]cnc3=N)C2)cnn2cccc(Cl)c12 C(CNC(c1n[nH]c(O)n1)=O)(C(=O)NCC(CC1CC1)CO)OC c1(CN=C(NCc2n(CC)ccn2)NC(C)C)ccc(F)c(O)c1 N1(C(C(CCC)OCC)=O)CC2(CCN2C(=O)CCC2CCC2)C1 N1(CN2C(=O)CN(C(=O)Cc3ccc(Cl)cc3F)CC2)CCCC2(C1)OCCO2 N1(Cc2onc(-c3cccc(OC)c3)n2)CC(NC(=O)CC2CCC2)CCC1C CC1CC(CNC(=O)CC2(O)CCOCC2)CCN1C(C1CC2CCC(C1)S2)=O CC1(C)CNC(CNCc2cnn(-c3ccccc3)n2)CO1 NC(=O)CCCC(=O)N1CCN(C(C2CCCCC23CC3)=O)CC1CCO C=CC1OCCC1NC(=O)C(C)N(C)C(c1ccc(N)cn1)=O CCCCC(CC)CC(=O)N1CCC(C)(C)C(C(=O)NC2CC(O)C2)C1 CCCCCC=CCC(=O)N(CCNC(=O)CNCC1CCCCO1)C1CC1 O=C(CCC(F)F)NCCC1CCCN(C(c2cccc(OC(F)F)c2)=O)C1 c1(C(N2CCCC(NC(CC(C)(C)F)=O)CC2)=O)cc(Br)c([N+](=O)[O-])s1 c1(C(N2CCC(C(F)(F)F)C(C)(C)C2)C(=O)NC)ccc2c(c1)CC(C)O2 Cc1cc(C#N)cc(C)c1C(N1CCCC1CCNC(=O)C(O)c1ccco1)=O c1(C(=O)NCC(C(C)C)(C)NC(=O)C(C2CCOCC2)C)coc2c1COC2 C#CCCC(O)C(=O)N1CCCC1OC(CNC(c1ccccc1)=O)=O CCC(CCCC(=O)NCC1(O)CC2CCCC12)c1ccccc1 C(CCCCC(=O)N1CCC(F)CC1C(=O)NCCCCCCCO)OCC C#Cc1ccc(Cl)c(C(N2CCCC(CNC(=O)C(C#N)CC)C2)=O)c1 n1(CC(=O)NC(C)CNC(=O)Cn2nccc2N)c(=O)cnc2ccccc12 N1(C(c2c(OC)scc2)=O)CCC(C)(NC(=O)COCCOCCO)CC1 N1(C2CC2)CCC(C(F)F)(NC(=O)S)C1.C1(CNC(=O)OC(C)(C)C)CC1(C)C.C N1(C(C(=O)NC(C)Cc2ccc(F)c(F)c2F)=O)CCCC1C1OCCO1 CCCCC(O)C(=O)NC1CCCN(Cc2cccn3ccnc23)CC1 C1(CNC(=O)COC(F)F)CCC(CNC(=O)C=C2CCCCC2)CC1 c1(OC)nc(Cl)ccc1CCC(N1CCCC1(C)Cc1cc(Cl)cc(Cl)c1)=O N1(C(c2ccc(CC)cc2)C(=O)NCCC2(C)CC2)CCOC2CCCC12 Cn1nc(C(=O)NC2CC(C(=O)NCCC(N)=O)C2(C)C)cc1O n1(CC)nnc(C(=O)NC(C)C)c1C.C1(C)CCN(C(=O)C(C2CCCCC2)C)C1 N1(C(c2cc(C)cc(Br)c2)C(=O)N(C)C)CCC(C2CCOC2)CC1.C1(C)C(=O)N1 Cc1cc(NC(c2coc(CNC(=O)CC3CC3CO)c2)=O)cc(CO)c1 C(=O)(CCS(N)(=O)=O)NC(C1CCCN(C(=O)C(F)(F)C2CCOCC2)C1)C C1(C)(CNC(C2CC(OC)C2)=O)CCCN(C(=O)CCc2c[nH]c(=N)[nH]2)C1 CC1C(NC(=O)C(F)(F)C(F)F)CC2CCC1N2C(c1cn2c(n1)CCC2)=O CC1C(NC(=O)C(C)(C)C2CCCCO2)CCN1C(=O)CC1CCOC1 CCC(CC)CC(=O)NCCC1(C(N2CCC(c3ncc[nH]3)C2)=O)CC1 N1(C(COC(CC)CC)=O)CCC(NC(C2CCC3(CCC3)O2)=O)C(O)C1 C1(C)(NC(COCC=C)=O)CC(NC(c2csc(C(C)(C)C)n2)=O)C1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC2C1 C1(CCO)(NC(C(C)SCCCC)=O)CN(C(=O)C(CO)c2ccccc2)C1 C(=O)(C(O)C(C)(C)C)NC1CC1N(C(C(c1c(OC)cccc1)C)=O)C12CC(C1)C2 C1(C#N)(C(=O)Nc2cccc(CNC(C(CCC)OC)=O)c2)CC12CCCC2 C1(CC(=O)Nc2cccc(C3CCOCC3)c2)CCCS(=O)(=O)C1 Cc1ccnc(C)c1NC(C1CCC(NC(=O)C(C)Cc2ccccn2)C1)=O CC(C)(C)CC(=O)NCC1CCC1CNC(=O)CN1CCCC(C(F)(F)F)C1 C1(C(N(C)CC2C3CN(C(=O)C=CC(C)(C)C)CC23)=O)CCCCCS1(=O)=O Cc1ccc(C)c(N(C)C(c2ccc(F)c(Cl)c2)=O)c1.C1(=O)C(C)N1 N(C(=NCCC1CC1)NC1CCS(=O)(=O)C1)Cc1n(-c2cn(C)nc2)nnc1Br C1(NC(C2(C)CC2)=O)CC2(CCN(C(C3CC(N4CCOCC4)C3)=O)C2)C1 CCC(C)C(C)C(=O)NCC1(NC(c2occ(C)c2C)=O)CCCCC1C C(=O)(C1NCCc2cc(C#N)ccc21)Nc1c(C)n(-c2ccc(Cl)cc2)nc1 C1(CNC(=O)CCn2cccc2)CC2CCC1N2C(=O)CCOCC(F)(F)F N1(C(c2ccc(C)[nH]2)=O)CCCC(C2CC2NC(=O)CCCCCc2cccs2)C1 C12(CNC(c3nnc(C)s3)=O)CC3CC(CC(C3)C1NC(C1CC(O)C1)=O)C2 C(=O)(CCCCCCBr)N1C(C(=O)NCCN2CCCC2=O)COCC1 C1(CCCNC(c2cscc2Cl)=O)CN(C(c2ccccc2C(N)=O)=O)CCO1 C1(NC(C2CC(=C)C2)=O)CN(C(c2ccc(N)cc2O)=O)CC1N=[N+]=[N-] c1(C(N2CCC(O)(CNC(=O)COC3CCCCC3)C2)=O)occ2c1CCOC2 c1(CC(N2CC(C(C)NC(c3c(C#C)c[nH]n3)=O)C2)=O)c[nH]c2cnccc12 N1(C(C2(C#C)CCCC2)=O)CCC2(CCC(CNC(C3CC3(Cl)Cl)=O)O2)CC1 N1(C(C2COC(C)C2)C(=O)NC(C)C)CCC2(O)CCOCC2C1 CCC(CC(=O)N(C)CC1(O)CN(C(=O)CC2(C)CCCCC2)C1)C(F)F C(CCCCC(=O)NC1CC1C(F)(F)F)NC(C1C(C)CC1)=O O=C(N=c1cc[nH]cc1Cl)C1CCCCC1C.c1(CN)cc(Cl)c(Cl)cc1O Cc1nc(Br)cnc1NC(C1(F)CCN(C(=O)C(C)(C)F)C1)=O Cc1c(NCCCc2ccsc2)ncnc1N1CCC(N(C)C2CC2)C1 C1(NC(C(C)CC2CCC2)=O)CCC2(CCCN2C(=O)CC(C)(C)C(F)F)CC1 N1(C(c2c(C)ocn2)=O)CCC(C2CCN(C(c3ccnn3CC(F)F)=O)C2)C1 CCCCCCC(C)C(=O)NC1CC(C)(NC(c2cncc(Cl)c2)=O)C1 N1(C(CCc2ccc(=N)[nH]c2)=O)CCCC(C2CC2NC(c2cnc(Cl)s2)=O)C1 Cc1nccc(C(N2CCC2CNC(=O)CC2(c3ccc(Cl)c(F)c3)CC2)=O)c1C C1(NC(CN(S(CC)(=O)=O)C)=O)CN(C(=O)OC(C)(C)C)C2(CCC2)C1 CCCC(C#N)C(=O)NC1CC(C(N2CC(F)(C(N)=O)C2)=O)CC1O N1(C(C(CC)F)=O)CCN(CCCNC(C2(C)CC(C)=NO2)=O)CC1 N1(C(=O)Oc2c(C)cccc2)C2CC1CN(Cc1ccnc(F)c1)C2 c1(SCC(=O)NCCC2(C(=O)NC3CCC(CO)C3)CC2)ccccc1 C1(NC(CCC=C)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 C1(C(N2CC(CCC)N(C(c3csnc3C)=O)CC2)=O)CCCN2CCCCC12 c1(C(=O)NCCC2CCCN(C(=O)C(F)C3CC3)CC2)ccc2nn[nH]c2c1 N1(C(=O)CCOCC2CC2)CCCC2(CCN(C(=O)CC3CC4CC4C3)CC2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)N1CC2C(N(C(C(C)OCC#C)=O)C)C2C1 Cc1nc(O)[nH]c1C(=O)NCC(C)(C)CNC(=O)C(c1ccc(Cl)s1)C c1(C(=O)NCC2CCN(c3nnn(C)n3)C23CC3)ccc2c(c1)nnn2C Cc1cnc(C(=O)NCC(C)(F)CNC(c2cc(C(F)(F)F)c[nH]2)=O)cn1 c1(C(=O)NC(CNC(C=CSC)=O)CC(C)C)cc2ccncc2[nH]1 C(=O)(CCCC(OC)OC)N(CC(N1CCC(CCC#C)C1)=O)CC c1(C(C)C)ccc(F)c(C(=O)NCC2CC2CNC(c2cccc(O)c2F)=O)c1 c1(CN(C(C2(CCO)CC2)=O)CC)c[nH]nc1C1CCN(C(=O)CC2CCOC2)C1 N1(C(C2(C(=O)OC)CC2)=O)CCC(C(=O)Nc2ccccc2SC)CC1.CCS CC1CN(C(=O)CC2C=CC(NC(c3ccc4[nH]ccc4n3)=O)C2)CC(C)(C)C1 N1(S(C(C)(C)C)(=O)=O)CC2CC1CC2c1ccccc1CO C#CCCC(O)C(=O)N1CC(C2CN(N)C2)C1.c1(N)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC(CCC)NC(C2COCCO2)=O)cc(F)cc(F)c1 N1(C(c2c(CC)cccn2)=O)CCN(C(c2cccn2C(C)C)=O)CC(O)C1 C#Cc1cc(C(N2CC(O)CC2C(=O)Nc2ccccc2CCO)=O)ccc1C N1(C(c2c(C)cc(F)cn2)=O)CCC(N(C)C(C2C(C)C2C)=O)C2(CC2)C1 C1(NC(C(Cn2ccnn2)NC(CCC(C)N(C)C)=O)=O)CCCN(C)C1=O C12(C(N3CCC(C(C#C)C)CC3)=O)CCCC1CCN2C(c1scc(C)c1C)=O N1(C(c2c(C)nccc2)=O)CCC(C)(C)C1C(N1CC(c2cc[nH]n2)C1)=O C1(C)(C(=O)NCC2(NC(CCC(C)(F)F)=O)CCOC2)Cc2ccccc2C1 c1(C(N(CCNC(=O)OC)C)=O)ccccc1S(C)=O C1(C(N2CCC(O)(CNC(=O)CCc3cc(Cl)cs3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(NC(=O)NC(c2ccc(C)cc2)C2CC2)c(C(F)(F)F)c1 c1(C(C(=O)NCCOCC)N2CCC2COCCOC)ncccc1Br C1(C(N2CC3CC(CNC(c4cccnc4)=O)C3C2)=O)CCc2ncsc2C1 N1(C(C2CCN(CC)CC2)=O)C2CCC1C(C(=O)NC1CC1(C)C)C2 C(C)(CCOC)NC(C1(N(C(C2(CCC=C)CC2)=O)C)CC1)=O c1(SC(C(=O)OC)COCc2ccccc2)cn(C)c2ccccc2c1=O C(CCC(N)=O)(C(=O)O)NCCC1OCCC(OCC)C1 c1(CC(=O)NC(C2CCN(C(COC(CC)C)=O)C2)(C)C)ccc(F)cc1F Cc1ncncc1C(=O)NC1CCC(CNC(=O)CNS(C)(=O)=O)CC1 c1(OC)c(F)ccc(F)c1C(=O)NC(C)CCCNC(C1(P(C)(C)=O)CC1)=O CC(C(C)(C)C)=CC(=O)NC1CC(NC(=O)C(C)(Cl)Cl)C1 Cc1cc(C)n(C(C)C(=O)NC2CCCC2(C)NC(=O)Cc2cncs2)n1 CN(C)S(=O)(=O)N1CC(C(=O)N(C)C(c2cccnc2)C2CC3CC3C2)C1 C1(NC(CCN(C(C2CCCC2CF)=O)CC)=O)CCN(CC)CC1 CCC(F)(F)CCN=c1nc2scnc2c(NCCSC2CCCCO2)[nH]1 OC1CN(Cc2cnn(CC3CC3)c2)CC12CCC2 C(=O)(CCS(C)(=O)=O)NCC1CCN(C(C(c2c(C)n[nH]c2C)C)=O)C1 c1(OC)ncc(CC(=O)NC2(CNC(c3cccnc3OCCO)=O)CC2)cn1 c1(C(=O)NCC2(F)CN(C(c3nc(C(C)=O)sc3)=O)C2)ccc2nc(C)oc2c1 n1(CC#C)ccc(N(C2CCCC2)C(=O)NC2CCOC2C(C)C)n1 C1(CCNC(c2cccc(C)c2C)=O)CN(Cc2nc(C(C)C)no2)CCS1(=O)=O N1(C(Cc2cn(CC)nc2)=O)CCCCC(NC(c2nn[nH]c2Cl)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC(C)C)CC2)=O)CC=CC1 c1(C(=O)NC2C(C)CCN(C(=O)CCC3CC3)C2)cc(F)c2c(c1)nnn2C C1(NC(=O)C(F)=CC2CC2)CN(C(C2CCC3(CCC3)O2)=O)C2CCCCC12 C1(C(=O)NC2CN(C(c3ccc(C(N)=O)s3)=O)CC2CO)CCCCC1C1CC1 N1(c2nc(N3CCC(C(NOC)=O)CC3)nc(C)c2)Cc2c[nH]nc2C(C)C1 N1(C(CC2=NN(C)C(=O)C2)=O)CCC(C2CCCN(C(C34CC(C3)C4)=O)C2)C1 C1(C(N(C(CC(=O)N(CC#C)CC2CC2)(C)C)C)=O)CCC(C)=C(C)C1 CC1CN(C)CCC1N(C(c1cc(Cl)ccn1)C(=O)NCC1CCCO1)C C(C(F)C(=O)NC1(CO)CN(C(C2COCC2C(N)=O)=O)C1)N(CC)CC N1(C(c2nnn(Cc3cc(C)no3)c2C)=O)CCC2(O)CCOCC2C1 c1(CN2CCC(CNC(c3ccc(OC)cc3)=O)CC2)ccc(O)c(C)c1 n1(CCC)cc(Cl)c(C(N2CC(NC(=O)C(C)(C)OC)C2)=O)n1 n1(CCC(=O)NCC2(C(C)(C)O)CN(C(C(CC)SC)=O)C2)c(C)csc1=O N1(C(c2cc(Br)co2)C(=O)NC(C(=O)OC)CC(C)C)CCC(C#N)CC12CC2 C1(C(=O)NCC(N)=O)CC2(CC2)CN1C(c1ccc(OC(F)F)c(F)c1)=O C(c1ccc2[nH]ccc2c1)=CC(=O)NC(C)CNC(c1cocc1Br)=O Cc1ccc(C(=O)N(C(C)(C(=O)N(C)CC2CCCCO2)C2CC2)C)c(C)n1 Cn1cc(C=CC(=O)N(CCCNC(C2(C(F)F)CCC2)=O)C2CC2)cn1 Cc1cc(F)ccc1CC(N1CCCC(CNC(C2CC(C(C)C)=NO2)=O)C1)=O C1(CNC(C(C(C)C)(C)C)=O)CN(C(c2ccnc(CO)c2)=O)CCC1(C)C Cc1cccc(OC(F)F)c1C.C12CC(C)(C)CN1N(C(C)(C)C)C(=O)C2.C(=O)O C(=O)(C(C)S(C)(=O)=O)N(C1CCN(C(C2CCCC(OC)C2)=O)C1)CC O=S1(=O)CC2CN(Cc3ccc(Br)c(Cl)c3F)CC2(C(F)(F)F)C1 CC1CN(C(C2(C)CCCS2)=O)CC1CCNC(c1nccnc1N)=O N1(C(CS(=O)(=O)NC)=O)CCN(C(C23CC(C2)C(C)O3)=O)CC1C CCCCC(CC)CC(=O)NCC1(F)CC(CNC(=O)CC2CCCC23CC3)C1 c1(C(N2CC(COC)(CNC(=O)CN(C)CCO)C2)=O)cnn2c1CCC2 N1(C(c2cnc(CC)s2)=O)CCCC(C)(C)C1CNC(c1ccc(O)nc1)=O C(CCCCCC(=O)NCCCC1CC1C)NC(C(C)OCCOCC)=O c1(-n2cc(C3C(OC)CN(C(C4CCCN(C)C4)=O)C3)nn2)ccc(F)cc1F c1(C(=O)NC(CCNC(C(C)OCC2CC2)=O)C)ncncc1N C1(NC(C(CC)N(C)C)=O)CCN(C(=O)CC2CC3(CCO2)CC3)CC(C)(C)C1 Cc1nc(O)ccc1C(=O)NCCC(C)N(C)C(c1cccc(CC2CC2)c1)=O N1(C(c2c[nH]c(=NC)o2)=O)CCC2C(C1)CN2C(=O)C(C1CCCCCC1)C CCC(C)CC(C(=O)NCC(F)CO)NC(=O)C(O)c1ccsc1 C1(CN(C(C=C2CCN(C)C2)=O)C)CN(C(=O)CSc2nccn2C)CCO1 Cc1nccc(C(=O)N(C)CCOCCNC(=O)CC2CCCCC2C)c1Cl c1(OC)ccc(C(CNC(=O)Cc2cnns2)NC(c2ccc(F)cc2)=O)cc1 Cc1cccc(C(N2CCCC2CNC(=O)CC2OCCCO2)=O)c1F c1(OC)ncc(CN2CCN(C(=O)Cc3cc(Br)cnc3O)CC2)c(OC)n1 N1(C(C(c2nccc(C)c2)(C)C)=O)CCCC2CN(C(=O)C(=O)NC3CC3)CC12 N1(CC)CCN(C(c2cc(OCc3ccccc3)ccc2O)C(=O)NC)NC1=O C(CS(=O)(=O)c1ccc(C(F)(F)F)cc1)NC(CC1(OC)CC2NCCC12)=O C1(C)(C(=O)OC)COCCN1C(=O)Cc1ccnc(C(C)(C)C)n1 CN1CC(NC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)CC12CCCC2 Cc1cc(O)n2ncnc2c1NC(=O)NCc1ccnc(OC(F)(F)F)c1 C#Cc1ccc(F)cc1C(=O)NC(CC)(CC)CCNC(C1(CCOC)CC1)=O N1(C(c2ccc(OCCN(C)C)c(Cl)c2)CC)CCN(C2CCCCC2)C(=O)C1 c1(-c2nc(CCCC)nn2-c2ccc3[nH]ccc3c2)ccc2nc(O)oc2c1 c1(C(C)C)ccc(C(c2nnnn2C2CC2)NCC2(CO)CCC2)cc1 c1(C(N2CCC(N(C(c3c(OC)cccn3)=O)C)C2)=O)ccnc2cc[nH]c12 c1(C(N(C(C)C(N2CCCC2CN(C)C)=O)CCC)=O)ccnc(OC)n1 CCC(C)C(O)C(=O)O.c1(N(CC(=O)N(CCCOC(F)F)CO)C)ccccc1 c1(N2CCC(C(=O)Nc3cccc(CC)c3)CC2)ncc([N+](=O)[O-])cc1Cl c1(OCC(=O)N(C(C)CC(=O)O)C)ccc([N+](=O)[O-])cc1 C1(C)(C(=O)NCC(c2ccccc2)NC(c2c(CC)cc[nH]2)=O)CCC(=O)NC1 C1(C(=O)NC(C(=O)N(CCCC)C(C)CC)(C)C)COCCC1C c1(C(N2CCC(N(C(c3cnc(COC)s3)=O)C)C2)=O)cccc(C(F)F)c1F c1(NC(C2CC(NC(c3ccc(Br)c(Cl)c3)=O)C2)=O)nc(Cl)ccc1O n1(CCNC(=O)NNC(=O)C2CCCO2)c(=O)oc2ccccc12 C12(C(N3C(C(=O)Nc4cccnc4)CC(O)C3)=O)CC3CC(CC(C3)C1)C2 C(=O)(C(C)CCCC(C)C)NCC1=CCN(C(CC(C)n2ccnc2)=O)CC1 c1(C(=O)NC2CC(C)N(C(=O)CCSC(F)(F)F)C2)ccc2oncc2c1 N1(C2CCCc3ccccc32)CC1.C1(C(=O)O)CC1(F)F c1(C(=O)NC2CCCC(NC(COC(C)C)=O)CC2)cnc2[nH]c(O)nc2c1 CC(C)C(O)C(=O)NC(CNC(=O)CCc1nnc(C2CC2)o1)C1CCCC1 c1(OC)ccccc1NC(=O)C(c1ccc(CCC(=O)OC)o1)N(C(C)C(C)C)C N1(C(c2c[nH]c(=NC)s2)=O)CCC(C)C(NS(=O)(=O)CCCF)C1 N1(C(C(C)NC(C2CCOCC2)=O)=O)CC2CC(NC(=O)Cn3ncnn3)C1C2 c1(CC(N2C(C(=O)NC3CC3(F)F)CC(F)C2)=O)c(Cl)cccc1Cl C=C1CC2(C1)CN(C(C1CCN(C(=O)CC(C)CN(C)C)C1)=O)C2 N1(C(c2cc(Br)c(C)s2)C(=O)NCCCCCC)CCC(O)C(F)C1 CCCCS(=O)(=O)N1CCCC1C(N1CCC1CNC(c1cnnc(O)c1)=O)=O N1(C(CC(=O)NCC)=O)CCCC2(C1)CN(C(C1(C)CCNC1=O)=O)CCO2 C1(N(C(c2cnc(CCC)s2)=O)C)CCN(C(=O)CCCCN(C)C)CC1C c1(C(=O)NC2C(NC(=O)C(c3ccc(Cl)cc3F)O)C2)csc2ccccc12 c1(C(=O)NCC2N(C(CCC(C)NC(N)=O)=O)CC2)ccc2c(c1)CCCS2 CC(C)(C(=O)NC1CC(CNC(C2CCCNC2=O)=O)C1)C(F)c1ccccc1 C(F)(F)(CN=c1ccc(Br)c(S(=O)(=O)N2CCC(C(N)=O)C2)[nH]1)C1(CC)CC1 Cc1cc(C(=O)NCC2CCN2C(=O)CCSCC(C)C)nn1C(C)C c1(C(=O)NCCCC(=O)N(C)C)cc2c(s1)CCN(Cc1ccc(F)cc1)C2 c1(C(N2C(CN(C)C(C3CC34CCC4)=O)CC(F)C2)=O)ccnc2c1CCC2 C1(C(=O)NC2CCN(C(c3onc(C)n3)C)CC2O)CC2(C1)CC(C)(C)C2 N1(C(c2c(COC)cc[nH]2)=O)CC(NC(=O)C(CCSC)N(C)C)CC12CCC2 N#Cc1ccc(C(F)(F)F)cc1S(=O)(=O)NCCNC1CCC(C(F)(F)F)CC1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2C3CCC2(C)C3(C)C)=O)C1 c1(C(=O)NCC(C)CNC(C2(C)CC2Br)=O)cc([N+](=O)[O-])n[nH]1 N1(C(CCNC(N)=O)=O)CC2CC3CC2C1C3NC(c1cn2sccc2n1)=O C(=O)(C1CCc2ccccc21)NC1CC(C)CN(Cc2ccc(Cl)cc2O)C1 N1(C(C=C(C)C2CC2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(NC(NOC)=O)ccc2c(c1)S(=O)(=O)N(C)C2=O N1(C(C(c2cn(C)nn2)NC(C(C(CC)C)=O)=O)=O)CCC2(CCOC2)C1 c1(C(=O)NCC2(CCNC(C3CC(CC(F)F)C3)=O)CC2)cc(O)cc(Cl)c1Cl N1(C(C(n2cc(-c3csc(C4CC4)n3)nn2)C)=O)CCC2(CCO2)CC1 c1(C(N(CCC#C)C)=O)ccc2c(n1)CN(C(=O)CC1CCCCC1O)CC2 Cc1cnc2c(C(=O)NC3CN(C(C4CC4(Cl)Cl)=O)CC3O)cnn2c1 N1(C(c2c(CC)nccc2)=O)CC2CCN(C(=O)Cc3ncoc3C)C(C2)C1 C1(CNC(c2ccc(Br)cn2)=O)COCCN1C(=O)CC1C=CCC1 N1(C(C2CC2C2CC2)C)CC(C)CC1C(N1CCC(n2ccnc2)C1)=O N1(C(C(C=CC)O)=O)CCCC2(C1)CN(C(=O)C=O)C2.c1(NC(C)C)ccc(S)cc1 c1(C(=O)NCCOC2CCN(C(C(CC)n3cncn3)=O)C2)c(C)noc1Cl C1(F)(C(=O)N(c2cc(O)cc(O)c2)C2CCOCC2)CCCN(C(=O)CCC2CC2)C1 C1(NC(C=C(CCC)C)=O)CC2CCC1CC2NC(C1(C)CCCC(F)(F)C1)=O c1(C(CC)CC)noc(Cc2cn(-c3ccccc3)nn2)n1 O=C(C1CCCn2cnnc21)NC1CN(C(c2nc(Cl)ccc2F)=O)C1 Cc1cnc(C2(NC(c3ccc(C4CCC4)s3)=O)CC2)o1.C1(=O)CNCCN1 N1(C(C)=O)CCCC2(NC(c3ccc(Br)s3)=O)CCCC12 C1(C(N(CC(C)(C)NC(=O)Cn2ncn(C)c2=O)C)=O)CC2(CCOCC2)CO1 c1(C(N2CC(CC(C)NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)ccc(F)c(C#N)c1 C=Cc1ccc(C(N2CC(NC(=O)C3=C(Cl)CCC3)C3CC23)=O)cc1 C1(CCNC(C=Cc2ncc(C)[nH]2)=O)CN(C(c2cscn2)=O)CCCO1 C(=O)(C(F)(F)CN1CCOCC1)NCC(CNC(c1conc1C(C)C)=O)OC CC1=C(C)CN(C(c2sccc2CNC(c2ccn(C(F)F)n2)=O)=O)C1 c1(C2N(C(=O)NCC(=O)O)CC2C)c[nH]c2ccccc12.C1(=O)C(F)(F)CO1 C=C(Cl)CCC(=O)N1CCC(c2nnc(CNC(C3(Cl)CC3)=O)s2)CC1 c1(C(N2CC3(CC(NC(CCC#C)=O)C3)C2)=O)cc(Br)c2[nH]c(C)nc2c1 c1(CN=C(NCC(COC)F)NC2CC2)nnc2cccnn12 C(=O)(C1=CC2CCC(C1)C2)N1C(C(N(C)CCc2nccs2)=O)CCCC1 CCCCS(=O)(=O)NCC(=O)Nc1cc(NC(c2ccccc2OC)C)n(C)c1 N1(C(c2cn(CC)nc2)=O)CCC(NC(=O)CN2CCCC2COC)C1C1CC1 N1(C(=O)NCCC(C)(C)SC)CC(CO)CC(C)C1 C1(NC(CN2CC(C)(C)C2)=O)CN(C(=O)CS(N)(=O)=O)CCC1O N1(C(C(C(C)C)O)=O)CC2C3CCC(C2C1)N(C(c1cccc2nonc12)=O)C3 C12(C(N(C3(CC(N4CCC=C(C)C4)=O)CC3)C)=O)CCCC1C2(F)F CCCC(C(=O)NCC#CCNC(C1(n2cccn2)CCC1)=O)S(N)(=O)=O C(CN=c1[nH]c(=NCCC(O)c2ccccc2)[nH]c2ccccc12)NC(C)=O Cn1ncc2c(NC3CN(Cc4ccc(Br)cn4)CC3(F)F)ncnc12 N1(C(C(CC)C)=O)CC(CO)C2(CCN(C(=O)Cc3c[nH]nc3O)CC2)C1 c1(C(N2CCC(NC(C(C=C)O)=O)C2)=O)ccc(-c2ccc(F)cc2)n1C C1(CNC(C2N(C(CCSCCC)=O)CCC2C)=O)CCCC(C)CC1 c1(C(=O)OC)nc(=NC2CC(F)(CNC(=O)C=CCO)C2)c(F)c(Cl)[nH]1 c1(C(N2CC3N(C(c4n(CC)ncc4)=O)C(C3)C2)=O)cc(Br)cc2c1cnn2C N1(C(CCc2ccn(C)n2)=O)CCCN(C(=O)CCC2CCC(=O)N2)CCC1 C(c1cc2ccccc2n1C)=CC(=O)NC(C)CC(C)NC(C1CC1F)=O c1(C(=O)NCC2CC(C)N(C(C3CCC3)=O)C2)nc2n(c1Cl)CCCC2 n1(C(CC)C)nnnc1C(c1ncc(I)s1)Nc1cnn(CCN(C)C)c1 c1(CC(c2ccccc2F)C)[nH]c(=NC(CCO)C(F)F)nc2c1cnn2C CCCCCC(C)(CC)C(=O)N1CC=CC(NC(=O)COCCC)C1 C(=O)(CC(P(C)(C)=O)c1ccccc1)NC(C1N(C(CCC)=O)CCC1)C Cc1ccc2c(C(=O)NCC(CO)NC(C3(n4cccn4)CC3)=O)coc2c1 C(=O)(C1=NOC(CNC(=O)CC(C)C)C1)NC(CC)(C)C Cn1cc2c(CN3CCC(O)C(C(=O)Nc4cccc(Br)c4F)C3)cccc2n1 Cc1cc(C(=O)NCCOCCCn2cc(-c3nc(C4CC4)cs3)nn2)sn1 O=C(CN=c1cc[nH]cc1)NC1CCCC(NC(=O)C(F)(F)C2(O)CCC2)CC1 Cc1c(C(=O)NC(C2CCCN2C(=O)C(C)N(C)C)C)cnn1CCO C=C(C)C(C)(O)C(=O)NC1CC(C(=O)NC2CCCCNC2=O)C1 c1(OC)cccc(C(=O)N(c2cnc(C(F)F)nc2)C)c1 Cc1cc(CNC(=O)CC2CCCC(C)C2)oc1C(=O)N(C)CC1(O)CN(C)C1 N1(C(c2ccc(C)cc2Br)=O)CCC2(CC1)CC(N1CCCC3(CNC3)C1)C2 c1(C(=O)OC)nn2ncccc2c1NCc1ccc(SCCCn2ccnc2)s1 c1(OC)cc(C(N2CC3CC2C3NC(=O)C(=Cc2ccco2)C)=O)ccc1C#N C1(C(=O)NCCNC(=O)NC)CCCN(C(c2ns[nH]c2=O)=O)C1 CCCC(CCC)CC(=O)N1CCC2CCC(C1)N2C(=O)CC(O)C(C)C C1(C(NOCCC(C)C)=O)CC2(CC2)CN1C(=O)CCCn1cccc1 N1(c2c(C)cncn2)CCC12CCN(Cc1ncc[nH]1)CC2 C1(C(=O)NC(c2ccnn2C)CC)CC(=O)CN1C(c1csnc1Cl)=O c1(N2CC(C)OCC2)[nH]c(=NCC23CCC(CC2)CC3)nc2scnc12 C1(CNC(c2ncn(CC)n2)=O)CC(F)(F)CN1C(c1cncc(C(=O)OC)c1)=O c1(CC(=O)NCCC2(NC(=O)C(O)CN3CCCC3)CCCC2)cccc(O)c1 C(=O)(CCN(OC)C(=O)C=Cc1cncn1C)NCC(N1C(C=C)CC1)=O.C(CO)OCCCC N1(CCNC(c2cnc(SC)s2)=O)CCC(NC(c2c[nH]nc2OC(C)C)=O)CC1 C(=O)(C(C)C1=CCCC1)NC1CCCN(C(Cc2nnc(C)s2)=O)CC1 c1(C(C)C)c[nH]nc1C(=O)NCCc1cc(C(N2CC(c3nncs3)C2)=O)no1 C(C)(C)(CC(=O)N(C)CC1CN(C(C2CC2c2nc[nH]n2)=O)CCO1)OC c1(C(N2CCCC(CNC(c3c(C)cno3)=O)C2)=O)ccc2c(c1)C(C)C(C)O2 Cc1ccc(CN(C)C(C2COCCC2c2ccccc2)=O)cc1F C(CCCC(=O)NC1CCCC(NC(c2n[nH]c(C)c2O)=O)C1)OCC C1(CC(=O)NCC(c2ccccc2)N(C(c2cc(C)[nH]n2)=O)C)SC(=N)NC1=O Cc1ncnc(C)c1C(=O)NC1CCC(C(=O)NC2CCCC3(C2)N=N3)CC1 CC1CCC(C(F)(F)F)N1N1CCC(O)(c2nc3ccccc3[nH]2)CC1 N12CCC(CC1)OCCOC(C)C2=O.C1(C)(C(=O)NC2CC2)CC2CC2C1 Cc1nc[nH]c1CC(O)C(=O)NC1COCC1CNC(=O)C=CC(F)(F)F C(=O)(CCCCCCS(N)(=O)=O)N(C1CCN(C(C2CCC(C)(C)C2)=O)C1)CC C1(n2cnnn2)CC2(C1)CC2CO.C(=O)(C1COC1)NC(C(N1CCSCC1)C)=O C1(C(=O)NC(CC(=O)OC)C)CN(C(=O)CCCCC2CC2)CCN1C c1(NC(C)=O)cccc(C(N2CCC(C)(NC(c3cnccc3Cl)=O)C2)=O)n1 C1(OC)CN(C(=O)CCn2ccnn2)C(C)(CNC(=O)CC2CCCSC2)C1 CC(C)C(C(=O)Nc1ccc2c[nH]nc2c1)C(C)NC(=O)Cc1cccnc1 C1(OC)CN(C(c2ccco2)=O)CC1NC(C1CCC(C(C)C)CC1)=O C#Cc1cccc(C(=O)NC(CNC(=O)Cc2ccc(Cl)cc2)C2CCC2)c1C N(C1CCOc2ccc(Br)cc21)C(=O)CC1COCCN1Cc1cccnc1O C12(C(=O)NCCC3(NC(c4cnn(CC5CC5)c4)=O)CCC3)CCC(CC1)CC2 C1(C(=O)OC(C)(C)C)(CCNC(=O)CC2(S(C)=O)CC2)CCOCC1 Cc1nc(O)ccc1C(=O)N(CC(C)CNC(c1cccc(O)n1)=O)C C(CCC(C)(C)C(=O)NCC1CCCOC1)NC(C1N(C)CCCCC1)=O C(C(=O)NC1CC(CCNC(C2(n3ccnn3)CC2)=O)C1)(C(C)C)NC(C)=O c1(C(N2CC(CC)N(C(C3CCC3CF)=O)CC2)=O)cc2c(s1)CCOC2 Cc1c(C(=O)NCCC(C)(C)NC(c2cccc(Cl)c2)=O)cc(Br)cc1N Cn1[nH]c(=NC(=O)C(Cc2ccccc2Cl)c2ccccc2)cc1Cl CC1CCCCC1(C)C(=O)NCC1CC(CNC(=O)Cc2c[nH]nc2O)C1 C1(NC(CC2(C=C)CN(C(C3CCC3(F)F)=O)C2)=O)CCN(C)CC1C#N N1(C(C=C(NC(C)=O)C)=O)CC2CC1CCC2NCc1ccc(NC(N)=O)cc1 c1(CC(N2C(C)(C(=O)Nc3c(C#C)cccc3)CCC2)=O)[nH]nc2c(Cl)cccc12 C=C(C(=O)N1CC2CC1C2CNC(c1c[nH]nc1-c1ccc(Br)s1)=O)C(F)(F)F C1(C(C)NC(=O)C(c2cncn2C)O)CCCN(C(c2nc(C(N)=O)co2)=O)C1 CC(C)(CC(=O)NCC1COC(C)(C)CN1C(c1ccc(N)cn1)=O)C(F)F CC1C(O)CCN1C(C1CN(C(C2C(C#N)C2(C)C)=O)CCO1)=O C1(NC(C2(C)CN(C(C(C)NC(C)=O)=O)C2)=O)CN(C(C)C)CC1C c1(C(=O)NC(C2CCN(C(C34CCC(C)(C3)OC4)=O)C2)C)cc2c([nH]1)CCCC2 Cc1ccc(C(=O)NCC2(CC(=O)NC(C)(C)CCN(C)C)CC2)c(C)c1 C(=O)(C(CNC(=O)COCCC(C)C)NC1CC1)NC(CC)C Cc1nn(C)cc1CCC(=O)NC(CNC(=O)CN1CC2CC2C1)C(C)C C(=O)(CCCC(C)CN(C)C)NCC(CC(C)C)NC(C1CCS(=O)CC1)=O c1(C(N2CCN(C(c3c(CC)ncnc3)=O)C(C)C2)=O)cncc2nc(C)[nH]c12 Cc1cc(N)cc(C(N2CC(C(C)NC(=O)CCc3cccnc3)C2)=O)c1F C(C)(CC(F)(F)F)N(C(CCn1c(C)ncc1)=O)C.C1CCO1 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC2CN(C(=O)CCc3cncnc3)CC12 C1(NC(C(CCC)CCO)=O)CN(C(=O)COCCCF)CC(C)(C)C1 c1(C(CNC(=O)C(C)SCC)NC(CCNC(CC(C)C)=O)=O)cccc(Cl)c1 c1(C2(NC(C3C(=C)C3)=O)CC2)nccc2ccccc12 Cc1nn(C)c(C(=O)NC(C)CNC(=O)C(c2ccc(F)cn2)(F)F)c1[N+](=O)[O-] Cc1cc(CC(=O)NC23CC(NC(=O)Cc4cc(C)on4)(C2)C3)cc(F)c1 C1(C(N(CC(=C)C)CC)=O)CC2CC1CC2NC(=O)CNC(=O)OC C1(C(N2CC(C#C)(N(C)C)C2)=O)CC(C)(C)CCN1C(=O)C(O)CCNC(C)=O C1(C(N2CC(C)C(CO)CC2)=O)CC2CN(C(=O)C(C)OC(C)(C)C)CC2C1 N1(C(CCc2ccc(SC)cc2)=O)CC2CCC1C(NC(=O)C(C)CF)C2 C1(CNC(C2OCCN(C)C2)=O)COCCN(C(c2cc(Br)on2)=O)C1 C1(C(N2CC(SCC)C2)=O)CCCC(NC(c2cc(CO)c(C)o2)=O)C1 C(c1cc[nH]n1)=CC(=O)NC(C(N1CCC(n2ccnc2)C1)=O)c1ccoc1 O=C(C1=C(Cl)CC1)NCC1CCN1C(=O)Cc1cc(Cl)sc1Cl C=CC1(CC(=O)NCC(C)C(=O)NC2CCC2)CN(C(C2(F)CC2)=O)C1 c1(C(=O)NCC2C(NC(CNS(NC)(=O)=O)=O)C2)cc2c(Cl)cncc2s1 C1(NC(c2n(CC)ccc2)=O)CCCC(NC(=O)Cc2cnn(C)c2C(F)F)CC1 c1(C(N2CCC(CCCl)CC2)C(=O)NCSc2ccccc2)cc(Br)ccc1Cl CC(C(O)C(F)F)NC(=O)CN(C(C1CC(C)(F)C1)=O)CC1CC1 CC1CC(NCC(=O)NC2CCC(C3CCCCC3)C2)CC(C)O1 C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C)C1CNC(C1Cc2nccnc2C1)=O c1(C(=O)NCC=C(C)C)cccc(CC(=O)NC2CC(NC(=O)C(C)C(C)O)C2)c1 CCC(C)CC(C(=O)NCCCCCC1CC1)NC(c1cocc1C)=O C(CCN(C)C)(C(C)(C)C)Sc1nccc(CNC(C(C)C#N)=O)c1 c1(OC)cc(C(=O)NC2(CCCCNC(c3cc(C)[nH]n3)=O)CC2)cc(C)n1 C12(CCNC(C3CN(S(CC)(=O)=O)C3)=O)CCC1CN(C(c1cc(C)co1)=O)C2 C12CCC3(CN(C3)C1=O)O2.C(CCCC(=O)N1CC(CC(C)(C)C#N)C1)OCC C1(C)(C(=O)NCC23CC(NC(c4c(F)ccc(C)c4)=O)(C2)C3)CCS(=O)(=O)CC1 c1(NCCN)ncc(OCC)cc1F.C1(O)(C(=O)C2CC2)CC(NC(C2CC23CC3)=O)C1 C(=O)(CC(C)(C)C(=O)NCCCCC(C)NC(=O)C(C)(C)C(O)CC)OCC C#CCCCC(=O)NCc1ccccc1CNC(=O)C(C)C(=O)OCC CCCCC(C)(F)C(=O)N(C(C)C(=O)NCc1cnc[nH]1)C c1(C(=O)OC)c(N2CC(=O)CC2)cccc1C.c1(-n2cccc2)cc(C)sc1C.OC c1(C(=O)NC(C(C)NC(C2C(COC)C2)=O)(C)C)oc2ccc(Cl)cc2c1C N=c1[nH]c(Cl)c(Cl)cc1C(N1CCCC(CNC(=O)CC2CNC(=O)C2)C1)=O C1(NC(c2n(CC#C)cnn2)=O)CN(C(=O)CC(C)(C)SC)C(C)(COC)C1 CON(CCC(=O)NC1CC(C)CCC1O)C(=O)C(F)C1CCCN1C N1(C(=O)C(O)C2CC2)CC(C2CN(C(C3CCC34CCC4)=O)C2)C1 c1(CC)cc(C(N2CCCC(NC(=O)Cc3cncn3C)CC2)=O)ccc1OC C1(N(C(c2cnc(CC)[nH]2)=O)CC)CCCCCC1.C(=O)C=CBr c1(C(N2CC(F)(C(=O)NCc3cncc(C#N)c3)C2)=O)ccnc2c1OCO2 N1(C(CCCSC(=N)N)=O)CCN(C(C2(C3CCCO3)CC2)=O)CC1 c1(C(N2CCCC(NC(c3ccc(Br)nc3Br)=O)C2)=O)cc(Cl)c(F)cc1F N1(C(c2cn(C3CC3)cn2)C(=O)NCC=C)CCCC2(CC2)C1 CC(CCCCNC(C1(O)CCOCC1)=O)NC(=O)C(C1CC1)N(C)C Cc1cc([N+](=O)[O-])ccc1NC(C)CCNC(=O)CCCCO C1(C(C)(C)C(=O)NCCCSCCO)CCCN(C(c2ccc(F)nc2)=O)C1 N1(C(c2ccnc(OC)n2)=O)CCN(C(C23CC(C)C2C3)=O)C(CC(F)F)C1 C1(NC(c2cc(C(C)(C)C)ncn2)=O)CC2CC(NC(=O)Cc3ccsc3)C2C1 c1(C(=O)NC2CN(C(C(C=C)(C)O)=O)CC2O)cnn2ccncc12 N1(C(C(CCC)OC)=O)CCCN(C(c2cccc(Cl)c2OC)=O)CC1C c1(C(=O)NCC(C(C)C)NC(C2CC=C(C)CC2)=O)cc(Cl)cc(Cl)n1 c1(C(N2CCC(NC(C3CC(F)C3)=O)C2)=O)cncc(C2CC2)c1 CC1(CNC(=O)CSCC(c2ccccc2)=O)CCN(C(=O)C(F)CC2CC2)C1 N1(C(c2c(CC)cco2)=O)CCC(F)(Cn2cc(-c3cncn3C)nn2)C1 C(=O)(CCCC(F)(F)F)NC(C1(O)CCN(C(c2cc3ncccn3n2)=O)C1)C O=C(N=c1cc[nH]cc1O)c1ccc(-c2ccc3nn[nH]c3c2)cn1 CC(C)CCC(C)N(C(=O)CN(C(C1SCCS1)=O)C(C)C)C C(=O)(C(F)(F)CCc1ccccc1)NC(C(C)C)(C)CNC(c1c[nH]c(=N)s1)=O c1(CC(N2CCC3(C(NC(CCSCC)=O)C3)C2)=O)c(C)nc(O)nc1O c1(C(N2CC(C)C(CNC(c3cc(F)cs3)=O)CC2)=O)cn2cccc(Cl)c2n1 N1(C(C(C(=C)Cl)(C)C)=O)CCC2CCN(C(c3ccn4c(C)cnc4c3)=O)C2C1 c1(C(=O)OC)cc(C(=O)NC2CCC(NC(=O)C(C)N3CCC3)CC2)c(C)[nH]1 c1(OC)cccnc1CNC(N1CCOCC1c1noc(-c2ccccc2)n1)=O c1(OC)ccc(NCCCN=[N+]=[N-])cc1.C12CCCN1C(=O)CSc1cnn2c1 c1(OC)cc(CC(=O)NC2CCN(C(c3cnn(C)c3C)=O)CC2C)ccc1F CCCCC(C(=O)N(C1CCCCCC1)CCNC(C1CC=CCO1)=O)C(C)C C(=O)(C1CCCn2ccnc21)N1CCC(OC)(CNC(C2CC3CCC2O3)=O)C1 N1(C(CC(C)F)=O)CCOC(C(=O)N(C2CCCCC2O)C)CC1 C1(CC(C)C)CN(CC(=O)NC2CCN(c3ncccn3)CC2)C(C)CO1 S(=O)(=O)(c1ccc2[nH]c(=NCC(F)F)sc2c1)N(CCC(C)O)C1CC1.CO Cc1cccc(C2=CCN(C(C3CC4CC4N3C(=O)COC(C)(C)C)=O)CC2)c1 C1(C(=O)NCc2c(CC)noc2C)CCCCCN1C(=O)C(C)NC(C)=O C(C(=O)NC(CC(C)C)C(=O)NCC1CCCCCC1)(C(C)(C)C)OC CC(C)CC(C)(C)C(=O)NCC(F)CNC(=O)Cc1ccc2nn[nH]c2c1 C1(F)(CNC(C(=Cc2ccco2)C)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 N1(C(C=C(C)CNC(=O)Cn2ccc(C)n2)=O)CCC2(C=CCO2)CC1 C1(O)(C(=O)NCc2ccccc2)CCN(C(C2CCC(F)(F)C2)=O)C1 c1(NC(C2C(OC)CN(C(c3cncc(O)c3)=O)C2)=O)cc(F)ccc1C C1(NC(=O)CCN2CCC(F)C2)CCN(C(=O)CCCCc2cnn[nH]2)CC1 c1(C(=O)NCC2(CNC(Cc3ccc(C)s3)=O)CC=CC2)c(C)ncn(C)c1=O c1(C(=O)NCC(C)CN(C)C(C2CC23CC3)=O)cccc(C2CC(F)(F)C2)c1 CC1CCC(CNC(C2CC3(C2)CC(O)C3)=O)CN1C(c1cc(C2CC2)[nH]n1)=O C1(C(C)C)CCCN(C(=O)Nc2cn(CC(N)=O)nn2)CC1 Cn1nc(C(=O)NCCC2(O)CN(C(=O)CC3CCC4CC34)C2)cc1Cl C12(C(N(CCN(C(=O)CC3CCC3)CC)CC)=O)CCC(C)(CO1)C2 c1(N2CCC(C)(NC(=O)CC(c3cccc(F)c3)O)C2)ncnc2c1CCC2 C1(C(N2CC(C=C)(CC(=O)NCCC(O)CO)C2)=O)CCCCCN1C C#CC1(C(N2CCCC(CCO)CC2)=O)CCN(C(=O)Cc2ccsn2)C1 C(CCCC(=O)N1CC(C(C(=O)NC(C)CF)OC)C1)OC c1(C(=O)NCC(C)N(CC(N)=O)C)ccc(C(F)(F)F)o1 N1(C(c2c(C)n(C)nc2)=O)CCCC(C)C1CCNC(=O)C=C1CCN(C)C1 N1(C(c2ccn(CCF)n2)=O)CCC(n2ccnc2)C1 C1(NC(c2c(CC)cc(Cl)cc2)=O)CC12CCN(C(=O)CCC(=O)OC)CC2 C12(C(N3CC4(CN(C(CCc5nc(C)c(C)[nH]5)=O)C4)C3)=O)CC1Cc1c[nH]nc12 c1(C(N2CC(O)(CCNC(CSCC(=O)OC)=O)C2)=O)cc(F)ccc1OC CCC(C)(C)C(=O)C(=O)NC1CCCC(C(=O)NCC(C)(C)NC=O)CC1 c1(CCC(=O)NCC2CC(O)CN2C(C2CC3CC2C3)=O)c(Cl)cccc1Cl c1(C(N2CCC(N(C(=O)CSC)CC)CC2)=O)cc2[nH]c(C(=O)OC)cc2o1 N1(C(C(C=CCCC)O)=O)C2COCC1CC(NC(C1CC(C(F)(F)F)C1)=O)C2 N1(CC(=O)NCC2N(C(c3c(C)nncc3)=O)CCC2C)CC(=O)N(C)C1=O Cc1noc(C)c1C(N1CCCC1CN(C)Cc1ccnc(Cl)c1)=O c1(OCC)ccc(C(=O)NCCCCCCNc2ncnc(O)c2Br)cc1C CC1(C)CCOC1C(=O)NCCC1(NC(C2CCCC2(F)F)=O)CCC1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(Cl)c1N N1(C(C2N(C(Cc3ccc(C#N)cc3)=O)CCC=C2)=O)CC2OCCOC2C1 C(C(C)(C)CCl)(c1n(CCCCCC)nnn1)NCCC(=O)N(C)C C1(CNC(C(c2ccc(Cl)cc2)C)=O)CC2CC2N1C(=O)CC1CSCCS1 CC1C(C)N(C(c2nn(C)cc2N)=O)CCN1C(C1CC2(CSC2)C1)=O CC(C)CCC(C(=O)NCCc1ncccn1)NC(c1cc(F)cc(F)c1)=O C12(NC(c3ccc(C)nn3)=O)CCOC(CNC(c3cscc3C)=O)(C1)C2 C(=O)(C(CO)C(F)(F)F)NCC1NC(=O)CN(C(c2nc(C)c(C)s2)=O)C1 CC(C)C(CC(=O)NC(C)(C(=O)OC)C1CC1)NC(=O)C(c1cnn(C)c1)C N1(C(C(C)NC(C)=O)=O)CC(C)(C)CC1CNC(c1ccc(C2CC2)c(F)c1)=O Cc1ccc(C(N2C(C(=O)NCCc3nncs3)CCC2C)=O)nc1 c1(C(N(CC(CC)NC(=O)C(C)(C)C2CCCCC2)C)=O)scnc1C c1(C(=O)NCC2(NC(C3C(OCC)CC3)=O)CCCC2)ccnc(S)c1 N12CCC3(CCCC3C1=O)CC2.C1(C(=O)NC2CC(OCC)C2)CCCC(=O)O1 C12(NC(c3c(Cl)nc(OC)s3)=O)CCN(C(=O)CCn3cccnc3=O)CC1C2 S(=O)(=O)(c1ccc(CNc2ccccc2)cc1)NC1C(O)CCC(C)C1 c1(OC)ccc2c(c1)CN(NCCC13CCC(C1)CS3(=O)=O)CC2 c1(CC)n[nH]cc1C(=O)NCCc1n[nH]cc1C(N1CCC(CSC)C1)=O N1(C(C2CCCCN(C(CC(=O)OC)=O)C2)=O)CCCC2CCCCC12 CC(C)C(C(=O)N(C)CCN(C)C)NC(=O)OC(C)(C)C.C12CCCN1C2=O N1(C(c2sccc2F)=O)CCC2CC2(C(=O)NC(C2CCCCC2)CO)CC1 N1(C(c2c(CC)ncnc2)=O)CC2CCC(CNC(=O)C(C(C)C)N(C)C)(C2)C1 c1(OC)ccc2cc(CN3CCC(C(=O)NCCc4cnn(C)c4)CC3)oc2c1 C1(NC(C2C3CN(C(C4CC=C(C)CC4)=O)CC32)=O)CC2CCC(C1)C2 C1(CC(=O)N(C(C2CCC2)C)CC)COCCN1C(c1ccc(CF)cc1)=O N(C)(C(=NCCC(C)=O)NCc1cc(N(C)C)ccn1)CC1CCN(CC=C)C1 C(C(=O)Nn1cnnc1C)(C1(O)CCC1)NC(CCCCCNC(C)=O)=O CC1CCCC(CC(=O)NC2CC3(C2)CC3C(=O)NCC2C3CN(C)CC23)O1 C1(NC(CCNC(COC)=O)=O)CC(C(=O)NC2CC3(CCOC3)C2)=CC1O N1(C(C2(C=C)CCN(C(=O)Cc3c[nH]nc3C)C2)=O)CC2(CO)CCC1CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)ccc2cc(Cl)ccc2c1 C1(NC(C(C)SC)=O)CC(CC(=O)NCCC23CC(CO2)C3)C1(C)C N1(C(C(C(C)(C)C)NC(CC(CC(=O)OC)C)=O)=O)CC(C)c2ncccc21 C1(C(C)NC(c2ccc(C(C)N)cc2)=O)CCCN(CCN2CCCCC2)C1 C1(NCCC(=O)NCCN(C)C(c2cccnc2)=O)CCCCCC1.C1(C(=O)N)CC1F C1(C(=O)NCc2ccc(COCC)o2)CN(Cc2ncccc2C)CC(=O)N1.CSC CC1CC(C(=O)NCCC(C)N(C)C(c2cc3c([nH]2)CCC3)=O)CC(C)(C)C1 c1(CC)ncc(C(=O)NC(CCNC(=O)C(c2ccc(Cl)s2)C)C(C)C)cn1 N1(C(c2c(C)nns2)=O)CCCCC1CCNC(=O)CCc1ccn(C)c1 C#CCCC(O)C(=O)N1CC(NC(c2c(Cl)cnn2C)=O)C(c2ccccc2)C1 N1(CCC(N2C(CN(C(C(C)SC(C)C)=O)C)CCC2)=O)Cc2ccccc2C1 C=C(C)CCCC(=O)NC(c1cccnc1)C(=O)NC(C)CCF N1(C(c2nc(CC)sc2)=O)CCCC(N(C)C(C2CC3C=CC2O3)=O)C1 Cc1cnnc(O)c1C(N1CCCC(CN=c2[nH]nc(C(N)=O)s2)C1)=O C#Cc1cccc(C(N2CCC2CNC(=O)Nc2ccc(F)cc2C)=O)c1 C(CCC(=O)NC(c1ccccn1)C)(C(C)C)NC(c1c(C)nncc1)=O N1(CCCC)CC(CNC(=O)Cc2cnn(C)c2Br)C(O)C1 C(N=c1[nH]c(=NCCCOCC)[nH]c2cccnc12)c1c(C2CC2)nn(CC)c1C c1(C(=O)NC(CNC(CC(=O)OC)=O)C)ccc(-c2ccccc2)c(C)c1 C1(C(=O)NCCN(CCOC)C(C2SCCCS2)=O)CCC2(CC1)CC2 c12ncncc1NC(c1ccccc1)CN(C)C2=O.C1(C(=O)OCC)(SC)CC1 CC(CN(C)C)CCC(=O)N(CC(C(=O)N1CCCC1C(O)CO)N(C)C)C1CC1 C(=O)(C1CCC(=O)c2ccccc21)N1CCN(C(c2ncn(C)n2)=O)C(CF)C1 CN1CCCC1C1CCCN1C(=O)Cn1cc(CCOCC2CCCC2)nn1 N1(C(c2ccc(C#C)o2)=O)CCC(O)C(NC(C2OCCN(C)C2=O)=O)C1 c1(NC(C2CC(O)CN2Cc2ccc(Cl)nn2)=O)ncc(Br)nc1Br c1(C(c2nnnn2CC(F)F)NCC2(COC)CC2)cn(CCO)cn1 C12(NC(c3c(CC)c[nH]c3)=O)CC3CCC(C1C2)N3C(=O)CCOC1CCC1 C1(CC)CCN(C(C2CCCC(CF)C2)=O)C1C(=O)NC C#CC1CC1C(=O)N(CCNC(C1CCC1CF)=O)CC CCC(C)CC(C)C(=O)N1CCC(CNC(c2cccc(OC(C)C)c2)=O)C1 C(=O)(CC(C)(C)C=C)N(CC(C)NC(C1CCCN1CC(F)(F)F)=O)CC CC1(C)COC(C(=O)NCC(C)(CO)NC(C2COCC2(C)C)=O)CO1 C1(CNC(C2(SC)CC2)=O)CN(C)CCN1C(c1cc(O)ccc1F)=O N1(C(c2ccncc2)=O)CC2CCC(C1)N(C(c1cc(Br)c(F)c(F)c1F)=O)C2 C(CCC(=O)NCC(CC)NC(=O)C(F)(F)C1(O)CCCC1)=CC C1(C(=O)NC2CN(C(C3C(C)(C)C3C(F)F)=O)C2)CCC2(C1)N=N2 CC(F)CC(=O)N.C(Cn1cncn1)(C(=O)N(CCC(O)CO)C)NC=O N1(C(C2CC(C)C2)=O)CC(C2CCCN(C(=O)Cc3cnc(O)nc3O)C2)C1 C=CCCCCCC(=O)NC1C=CCN(C(=O)CCOc2ccc(Cl)c(Cl)c2)C1 C1(CNC(C2CSCN2C(CCOCCO)=O)=O)CCOCC1 C=CCC(CC(C)C)C(=O)NCC1(NC(=O)CCc2ncccc2C)CCC1 c1(C(N2CC3CC3(C(=O)Nc3ncc(F)s3)C2)=O)c(C(F)(F)F)cccc1Cl Cc1c(C(N2CCC(O)(C(C)NC(=O)CN3CC(C)C3)C2)=O)sc2nccn12 c1(CNCC23C(CN(C(c4cc(C)[nH]n4)=O)C2)C3)c(Br)cc(Br)c(O)c1Br C12(C(N3C(CNC(C4N(C(C)=O)CCCC4)=O)CC3)=O)CCC(C)(C(=O)O1)C2(C)C c1(NC(N2CCCC(NC(CC#C)=O)C2)=O)cccc(Br)c1O c1(CNC(C2CC(OC)CN2C(C2CCN(C)C2)=O)=O)c[nH]c2cnccc12 C12(COC)CN(C(=O)CCCn3cncn3)C(CNC(C3CCOC3)=O)(C1)C2 N1(C(C(=O)NCC2N(C(C(CC)O)=O)CCC2)C)Cc2ccccc2C1=O N(C1CCCc2nn(C)cc21)S(CC(C)c1cccc(Cl)c1)(=O)=O C(=O)(CC(C(F)F)N(C)C)NC1CCC(CCC(=O)NCc2c(C)nccn2)C1 C1(NC(COCCCOC)=O)CCC(O)CN(C(=O)C(N2CCNC2=O)C)C1 c1(C(=O)NCC(CC)NC(C2C3CCOCC23)=O)cn(C)nc1C1CCCC1 c1(C(=O)NC2(C(=O)NC(c3ncc[nH]3)CC)CCC2)cc(C(F)F)cs1 C1(C(N(CCCNC(=O)CC2CCCC2C)CCC)=O)CC(F)(F)C1(C)C C1(C(N2CCC(n3[nH]c(C4CC4)nc3=O)CC2)=O)(SC)CC(F)(F)C1 CCCCCC(C)(CC)C(=O)N(CCCN(C1CCN(CC)CC1C)C)C C1(O)(CC)CCN(C(c2ccnc(CNC(c3cc(C(N)=O)[nH]n3)=O)c2)=O)C1 CCC(C)C(O)C(C)C(=O)NC(c1ccccc1)CNC(=O)CCCC(C)(C)C c1(C(N2CC(C(N)=O)(CNC(C3C(C)(C)CCC3)=O)C2)=O)nc2ccccn2c1F c1(C(=O)NCC2N(C(C(C)OCCC=C)=O)CCC2)ccccc1[N+](=O)[O-] C(F)(C(=O)NCCC1CC(NC(=O)C(C)n2cnnn2)C1)OC C1(NC(CSCC(=O)OC)=O)CC2(CCN(C(c3ccns3)=O)C2)C1 C1(NC(C2CCC(CC)O2)=O)CC12CCN(C(=O)C(C)=C1CCCC1)CC2 c1(NC(C(c2cnc(C)[nH]2)N(C(CCO)C(F)(F)F)C)=O)cccc(Cl)c1C C12(C(N)=O)CCCC1(C(N1CC(CO)(NC(C3CC3F)=O)C1)=O)C2 N1(C(C(CO)NC(c2c(C)n(C)cn2)=O)=O)CC2CC3CC2C1C3 S(=O)(=O)(c1cccc(C(N2CCC(F)C(NC(=O)C3CC3)C2)=O)c1)NC C(=O)(CC1=NNC(=O)C1)N1CCOCC(CNC(=O)COCC2CCC2)C1 C1(C)(C(N2CC(CC(=O)NCC(C(C)C)O)OCC2)=O)C(C)(C)C1(C)C C(N=c1ccn(CC(N2CCC3(CC2)CC3)=O)c(O)n1)c1c(OC)cccc1 C=Cn1nccc1C(=O)NC1(CCNC(C2ON=C(C)C2C)=O)CC1 C(CC(F)F)(C(=O)NCCN1CC2CC2C1)NC(c1nnn(C)c1N)=O CC1CC(=O)NC(C(N2CCC(C)C(CC(=O)NCCC(O)C(F)F)C2)=O)C1 C1(NC(C2C(CC)OCC2)=O)CC(C)N(C(=O)CC2CC3(CCC3)C2)C1 c1(NC(N2C(c3ccc(C(=O)OC)s3)CCC2)=O)ccc(F)c2[nH]ncc12 C1(CNC(CCSCC(=O)OC)=O)CCCCN1C(=O)CCCC1CCCC1 C1(C(=O)NCCNC(c2nccc(CC)c2)=O)CC2CCCC(C1)C2=O C=C=CC(C)C(=O)N1CCC(O)(CN(C)C(c2ccc(OCC)cc2)=O)C1 CCCCCC(C)CC(=O)NCCOCC(N1CCCCCC1C(C)C)=O N1(C(c2c[nH]c(=NC)o2)=O)CCC(C)(C)C1C(=O)NC(c1ncc[nH]1)CO C1(CC(=O)NC2(C=C)CCC2)CCN(C(=O)C(F)=CCC)C1(C)C C1(C(N2C(CN(C(c3nc(CC)oc3)=O)C3CC3)CCC2)=O)C2CCCC(=O)C12 C1(C(=O)NC2CC(C)(CNC(C3CC(O)C3)=O)C2)CCCC(C)(C)CC1 N1(C(C(CC)NCC)=O)CCC2CN(C(C3CCN(C(=O)CC)C3)=O)CC2C1 C1(C(N(C)CC2CCCC2)=O)CC12CCN(C(c1cnc(O)c(F)c1)=O)CC2 c1(C(=O)NCC2(NC(c3ccc(C(C)=O)nn3)=O)CC2)ccc2n[nH]cc2c1Cl c1(C(=O)OC)ccc(F)c2c1CN(Cc1cccc3sc(O)nc13)CC2 N1(C(C(CC#C)C)=O)CCCC2CN(C(C3CC(SC)C3)=O)CCC12 C1(SC)CN(C(c2ccc[nH]2)=O)CC1NC(c1nn(C(C)C)nc1Br)=O N1(C(C2CN(CC)C(=O)C2)=O)CC(NC(=O)CC(C)C)CC12CCCC2 N1(C(c2ccc(OC)s2)=O)CC(CNC(c2sccc2OC(F)F)=O)CCC1C C1(CNC(C(CC=C)(C)C)=O)CN(C(c2ccc(CC)[nH]2)=O)CCC1(F)F CCC(CC(F)(F)F)C(=O)N(CC(C)NC(C1CC2(C1)CC(C)(C)C2)=O)CC N(C1CN(C(=O)CSc2nc[nH]n2)Cc2ccccc21)C(c1c(C)cn(C)c1)=O CC1(C)CC(C(=O)NC2COCC2C(=O)NCCOc2ccncc2)CCO1 C(=O)(C(C)C(C)n1cccn1)OC(c1c(C(N(CC(=O)NC)C)=O)nns1)=O C=CCC(C)(C)C(=O)NC1CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 c1(OCC)ccc(NC(C2CN(C)CCN2C(C2(F)CCCC2)=O)=O)cc1C C(C1c2ccccc2CCN1C(=O)C1=CCSC1)NC(c1c(C)cccc1)=O N1(CC2CCCC(CC)C2)CCc2nc[nH]c2C1c1ccc(F)cc1 C1(CC(=O)OC)CN(C(=O)NC2(CO)CCCCC2)CCCO1 N1(C(=O)CC2CCCCC2)CCC12CN(C(C1(c3ccccc3)CCCC1)=O)C2 CC(C)CC(C(=O)NCc1cc(OC(C)C)no1)NC(=O)C(C)(C)Cl C(C(=O)N=S(C)(C)=O)NC(c1ccncc1C)c1n(CCSC)nnn1 C=CC1CCCN(N2CCN(c3nc(C(C)(C)C)nc(C)c3C)CC2)C1 CC(C)(C)C(O)C(=O)NCC1(O)CC(NC(C23COC(CS(C)(=O)=O)(C2)C3)=O)C1 C1(C(N2CC3C(CNC(=O)CCC4CCOCC4)(C3)C2)=O)(CF)CC2(CCC2)C1 c1(C(=O)NC2COCC2NC(C2(CF)CC2)=O)cccc(CC2CC2)c1 CC1(C)COCCC1C(N1CCC(CCN)CC1)=O.c12csc(n1)CNC(=O)C2 CC(C)(C)C(C#N)C(=O)NC1CC(O)(CNC(c2ccc3ncnn3c2)=O)C1 N1(C(C=C(COC)C)=O)CCC(NC(=O)CSC2CCCCO2)C1C1CC1 C12(C(N3CC(CNC(C(CC=C)N(C)C)=O)(OC)C3)=O)CCC(CC)(C1)OC2 C1(CO)CN(N2CCCC2Cc2cccc(F)c2F)CCO1 C1(C)(CNC(CCC2(C)CC2)=O)CC(F)(F)CN1C(c1cccc(Cl)c1O)=O C1(C(C)C)CN(C(C2COCC2NC(C2CCC3CC2CO3)=O)=O)CCCO1 C1(CC)CCCN(C(C2CCC(C(N)=O)C2)=O)C1C(N1CCN(C(C)=O)CC1)=O N1(c2nc(N3CCC(CCO)C3)cc(C)n2)CCC2(CCCCO2)C1 C(=O)(CC(CC)N(C)C(C1(CC)CCCN1C)=O)NC(C=C)C N1(C(CCN(C(C)=O)C)=O)CCCCC1CNC(C1CC(CC2CC2)C1)=O C1(CC(=O)NC2CN(C(C(CC)N(C)C)=O)C2)CC(=O)NC(=O)C1 C1(NC(C(CC)CC)=O)C2CCN(C(=O)CC3CCCO3)CC12 c1(C(N2CC(C(C)NC(C3CCC3n3ccnc3)=O)C2)=O)cc(Cl)c(Cl)n1C C1(NC(C(C)(C)CC#N)=O)CCC2(CC1)CCN(C(c1conc1C1CC1)=O)C2 c1(CNC(C=C(C)C)=O)ccc2c(c1)CCC2NC(=O)C(F)(F)c1nccs1 CCCC(C(=O)N1CCC(N(C(c2cc(C)sn2)=O)CC)CC1)NC(C)=O C(=O)(CC(C)C(=O)OC)NCCC1CCN(C(C(CC)CC)=O)C1 C=C=CCCC(=O)NCC1CCC1NC(=O)C(N1CCOCC1)C1CC1 c1(CC)[nH]nc(C(N2CCC(O)(CN(C(=O)C(C)C#N)C)C2)=O)c1Br c1(OC)c(F)cc(C(=O)NCC(CNC(C2CCC(C)(C)C2)=O)CO)cc1Cl c1(CCN)noc(C)n1.C1(C(=O)NC)CC1C(F)(F)F Cc1csc(=NCC(=O)NC2CC(F)(CNC(c3csc(C)n3)=O)C2)[nH]1 c1(C(N(c2ccc(C)cc2)CCC#N)=O)cc(O)cc(=O)o1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCC1(CNC(=O)CCCS(N)(=O)=O)CC2 N1(C(C(C=C)O)=O)C2CCCC1CC(NC(=O)Cc1ccccc1S(C)(=O)=O)C2 c1(N(CCN2CCC(c3noc(C)n3)C2)CC)ccccc1C CCC(C)C(CC(=O)NOCCC(C)O)NC(=O)C#CC(C)C CC(C(C)C(=O)NCC1(CNc2ncccc2[N+](=O)[O-])CCCC1)S(C)(=O)=O N1(C(C2C(C(C)O)C2)=O)CC(CNC(C2CC2(C)C)=O)C1 c1(C(=O)NCC(C(=O)NCc2ccnn2C(C)C)OC)cccc(Cl)c1 N1(C(C(N2CCC(C)C2)=O)=O)CCCC(O)(CNC(=O)C=CCN2CCCC2)CC1 C12CCC(CC1)NC(=O)CC1CC(C1)NC(=O)C2.C(C(C)C)N(CC)CC c1(C(=O)NC2C(CNC(COCCC=C)=O)CCC2)ccncc1Br N1(C(C(N2CCN(CCCC(C)O)CC2)=O)=O)CC2CCC(O)C(O)C12 c1(N2CC(CNC(C(c3cncnc3)C)=O)OCC2)ncc(C#N)cc1Cl N1(C(CC(CC)O)=O)CCC(NC(c2c(C)coc2C(C)(C)C)=O)C(CC)C1 C(=O)(C(CNC(=O)COC1CC(NC(=O)CCCc2ncco2)C1)OC)OC C1(F)(C(=O)NCC2C(C(NOCC3(C)CC3)=O)CCO2)CCOCC1 Cc1ccc(C2(C(=O)NCC3(CC4CC4)CC3)CC2)cn1.C12CCCCN1C2=O N1(C(C(F)=CC)=O)CCC(CNC(c2n[nH]cc2-c2ccccc2)=O)C(C)C1 C(=O)(C1CCc2c[nH]nc21)NCCC(C(=O)NC1CC(C)(C(N)=O)C1)OC N1(C(C)C)CC(C(N2CCC(CNC(c3ccnn3C(C)(C)C)=O)C2)=O)CC1=O Cc1nn(C)cc1C(=O)NC1CN(C(c2nocc2C)=O)CC1C C1(CNC(C(C)(CO)NC(C)=O)=O)CN(C(=O)COC(=O)OC(C)(C)C)C(C)(C)C1 C12(CCCC1C)C(=O)N2.c1(C(=O)NCc2c(C)nsc2)cc[n+]([O-])cc1 NC1COC2(C(N3CCCC(C(c4nc(C5CC5)no4)O)C3)=O)CC1C2 C(=O)(C1CCCc2ncnn21)NCCC1(NC(=O)CCC2CCOC2)CCC1 c1(C(=O)NCC(C)NC(=O)C(O)CF)cc(C(F)(F)F)ccc1[N+](=O)[O-] C=C(C)CC(C(=O)N(C(C)CSC)C)NC(c1ncoc1CC)=O C1(C(N)=O)CN(C(C2CCCC2NC(=O)C#CC2CC2)=O)CC12CC2 C1(C(=O)NCCC2CCCC2(F)F)(CNC(=O)OC(C)(C)C)CCOCC1 c1(N(C2CCOCC2)C)nc(=NCC2CCC2(F)F)[nH]c2c(F)cccc12 C(=O)(C1=CCCCCC1)NC(CC#C)C(=O)NCC(C)(O)C(F)F C(N=c1[nH]c(=NCCCN2CCC(O)C2)c2ncccc2[nH]1)c1n(C(C)C)ncn1 c1(C(=O)NC2C(C(=O)Nc3c(C)ncnc3)C2)c(F)cc(C#N)cc1F N1(C(CCCOC)=O)CCC2(CC1)CN(C(c1ccc(F)c(C)c1)=O)CC2CO C1(CNC(CN(C(=O)CSCC(F)(F)F)CCOC)=O)CC1(C)C C(=O)(CC(C)(C)CNCC(C(C)NC(=O)C(C)N(CCO)CCN(C)C)(C)C)NC c1(-n2ncc(C(N(CC(CNC(C(CC)(C)C)=O)O)C)=O)c2)ccc(F)cc1F N#Cc1ccc(CNC2(c3nnnn3CC(F)F)CCNCC23CC3)cc1F C1(NC(C2C(=C)C2)=O)CCC(CN(C(=O)CCCc2cnccn2)C)CC1 C1(NC(C2(CC(C)C)CCC2)=O)CC=CCC1OCC.C1C(C)NC(=O)O1 c1(OC)cc2c(cc1CN1CCC(CO)(CO)CC1)OCO2 c1(C(C)=O)ccc(Sc2cccc(NC(c3oc(C4CC4)cc3C)=O)c2)cc1 C(C(CC(F)(F)F)NC(C1CC(=O)NC1(C)C)=O)NC(C(CC)=CC)=O N1(C(CCCC)=O)CC(CC2(C(=O)OC)CCCO2)C(F)(F)C1 O=S(=O)(c1cccc(N2CCOC(C(F)F)CC2)n1)NCCCOC1CCCC1 N1(C(CCC2(C)CN(C(CCCOC(C)=O)=O)C2)=O)CC2(CCN(C)CC2)C1 C1(S)C=CCCC1.C(C(C)C#N)N(CCNC=O)CC.C12(CCC1)CC(=O)N2C1CC1 C=C1CC(C(=O)NC)(CCCNC(=O)CC)C1.C(C(C)C#N)C(=O)N c1(C(N2CCC(C(F)(F)F)CC2)C(=O)NC)ccc(OCC(C)C)nc1C C1(CC(C)C)CN(C(=O)CN(C(=O)CN(CCC(C)C)C2CC2)CC2CC2)C1 C1(NC(NCC(C(C)C)OC)=NCC2CC2)CCn2c(C(F)(F)F)nnc2C1 c1(CNC(C(C(C)OC)NC(=O)CC2CNC(=O)O2)=O)nn(C)c(=O)n1C CN1CCC(C(=O)NC2CCC(CNC(c3cnc[nH]c3=N)=O)CC2)C1=O C(=O)(CC(C(F)(F)F)n1ccnc1)NC1CC(CNC(C(C)OCC2CC2)=O)C1 N1(C(c2c(C)cccn2)=O)CCC(NC(C2CCC(=O)N2)=O)C(CO)CC1 c1(OC)ccc(-c2ccc(CN3CC(NC(C4CCN(C)CC4)=O)C3)cc2)cn1 c1(NC(c2cnn(-c3ccc(O)nn3)c2C(F)F)=O)nc2ccccc2o1 Cc1ccc(C(=O)N(CC(C)N(C(=O)CCn2cncn2)C)C)c2cccnc12 c1(OC(C)C(=O)N2CCC2CNC(=O)CCC2CCCO2)ccc(F)cc1 C(=O)(C1CCC(=O)c2cccn21)N(C(CNC(C=C(CCC)CCC)=O)C)CC c1(CC)onc(C)c1C(N1CCC1CC(=O)N(C1(N2CCOC2=O)CC1)CC)=O C(=O)(C1=C(C)CCOC1)N1C(C(=O)NC2(CC=C)CCOC2)CC(F)(F)C1 C(C(C(=O)N(CCCOCCNC(C1CC1C)=O)C)C(F)(F)F)OC c1(C(=O)NCC2C(CNC(c3c(CC)nns3)=O)C2)cc2c(O)cc(Cl)cc2[nH]1 CC(N=c1nc2c(cnn2C)c(NCc2ccc(C(F)(F)F)o2)[nH]1)C1CC1 N1(CC)N=C(C(=O)N2CC=CC2CNC(c2cnco2)=O)CCC1=O Cc1nccc(C(=O)NC23CC(NC(=O)CC4CCCN(C(C)C)C4)(C2)C3)c1Cl CC(C)CS(=O)(=O)CC(=O)N1CCOCC(CNC(=O)C2=CCOCC2)C1 C1(N(C(=O)Cc2cn(C)cn2)C)CCN(C(c2cccc(N)c2F)=O)CC12CC2 CC12CCOC(CNC(C3CC(O)CCN3C(=O)COCC3CC3)=O)(C1)C2 C1(OC)CC2(CCN(C(C3(C)CC(O)CN3C(c3coc(C)c3)=O)=O)C2)C1 C1(C(C(=O)NCC(CCNC(CCSCCCC)=O)OC)C)CCCCCC1 C(C(COC)C(=O)NCC1(C(C)(C)C)CCN(C(C2CC23CCC3)=O)C1)OC Cc1ccccc1CC(=O)N(C(C)(C)CC(=O)NCCN(C)C1CC1)C C1(CNC(C(C2CCC2)OC)=O)CN(C(=O)C(F)=C2CCC2)C2(CCC2)C1 c1(C(=O)NC2CC(O)(CO)C2)cccc2ccc(Br)nc12 Cc1c(C(N2CCCC(C)(CNC(C3CSC3)=O)C2)=O)cnc2ncnn12 C1(c2cn(C(C(N3CCN(C)CC3)=O)N)nn2)CC2(CCCN2)C1 Cc1ccc(F)c(CS(=O)C(C)C(=O)N(Cc2ccccn2)CC2CC2)c1 C(=O)(C1=CCC(C)CC1)NC(CCCNC(c1c(CC)ncnc1)=O)C CC(=O)C(C)(C)CC(=O)N1CC(CO)(NC(=O)C2=CCCS2)C1 N1(C(c2c(C)oc(Cl)n2)=O)CCC2OCCN(C(=O)CS(=O)(=O)N(C)C)C2C1 N1(C(CSCC)=O)C2CCCC1CN(C(C1Cc3ccccc3C1)=O)CC2 c1(C(N2CCC(OC(CNC(=O)NC)C)C2)=O)cccc(NC(C)=O)c1 N(C(=NCCCF)NCC1CC1)CC1CN(C(=O)OC)C1.C1CCS1 C1(CNC(=O)Nc2c(OC)cc(C)cc2)CC2CCC1N(C(=O)CC1CC1)C2 c1(CC(=O)NC(CC=CC(=O)NC(c2ccn(C)n2)CC)(C)C)c(C)noc1C C12(NC(CCc3cnc(C)o3)=O)CCCCCC1N(C(=O)CSCC(N)=O)CC2 C1(C(=O)NC(CN2CCN(C(CC(CCC)O)=O)CC2)C)CCc2nccn2C1 C(c1c[nH]c(=N)c(C)c1)=CC(N1CC(NC(c2[nH]cc(C)c(=O)c2)=O)C(C)C1)=O C#CC1CCCN1C(=O)C=CCN(C(=O)C(CC)CC)C c1(OC)nccc(C(=O)NCC#CCNC(c2ccsc2Cl)=O)c1F N1(C(C(C)CC(F)F)=O)CCC2(C1)CN(C(C1CCC(F)(F)CC1)=O)CCO2 c1(C(N2CC(NC(c3cnn(CC)c3Br)=O)C(O)C2)=O)ccc2c(c1)CC2 Cc1[nH]nc2ccc(C(=O)NC(C)C(C)(C)NC(C3CCCCCC3)=O)cc12 C1(C(F)(F)F)(N(CCN(C(c2ccncc2Cl)=O)CC)C)CCCCC1.CC N1(CC2CCC(NC(c3cc(O)nc(COC)n3)=O)CC2)CCc2n[nH]cc2C1 C(=O)(C#CC1CCCO1)N1CCC(CNC(Cc2c(OC)nccc2)=O)(OC)C1 C1(OC)(CNC(c2ccnc(O)c2)=O)CCN(C(c2ccsn2)=O)CC1 C1(C(=O)NCc2cnccc2Cl)CCC(C(=O)Nc2ccc(O)nc2)CC1 C(=O)(C1Cc2ccc(C)cc21)NCCNC(CCCC)=O CCCC1C(=O)NC(C(=O)N(CC)CC2CC3CCC2C3)CO1.C(C)(C)OCC C12(NC(C(C)(C)CF)=O)CCC(CNC(=O)Cn3nc(O)ccc3=O)(CC1)OC2 N1(C(c2c(F)ccc(OC)c2)=O)CCN(C(=O)CNC(N)=O)CC(C)C1 Cc1cc(Cl)cc(N)c1C(=O)NC1CCN(C(=O)C(C)CC(F)(F)F)C1 CC1CC(NC(=O)CSC)CN(C(c2ccc(NC(=O)C3=COCC3)o2)=O)C1 C=CCC(CNc1c(C)ccnc1OC)C(=O)OC C1(NC(CC2N(C(Cc3ccc(C)o3)=O)CC2)=O)CC12CCCC2 N1(C(COCc2cccc(C)c2)=O)C2CCC1CC(NC(C1CCC=CO1)=O)C2 C1(CNC(Cc2c(C)ocn2)=O)CC(C(=O)NC(CO)CCN(C)C)=NO1 C1(C(N(C2CN(C(c3cnc(SC)s3)=O)CC2O)C)=O)CCc2nnc(C)n2C1 c1(C(=O)NC2C(CNC(c3cc(CC)on3)=O)CC2)ccc(=O)n(CCOC)c1 C1(C2CN(C(C3CC3C(F)(F)F)=O)C2)(NC(Cc2cn(C)nn2)=O)CC1 n1(CC)ncc(Cl)c1C(=O)NCC(F)CNC(=O)CC(C)n1ccc(C)n1 C(c1cccc(Cl)c1)=C(C(=O)NCC1CCN(C(c2c(C)nc(OC)s2)=O)C1)C c1(OC)cc(C(=O)NC2CC2CNC(=O)COc2cccc(O)c2)cc(Cl)c1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CCCN2C(C2CCOC2(C)C)=O)C1 c1(C(=O)NC2CCCC(CC(=O)NC3(CN(C)C)CCC3)C2)ncc(F)cc1F C12(C(N3CCC(C(C)NC(C4CCN(C)C4)=O)CC3)=O)CCC(CC1)CO2 CN1CCCC1CCC(=O)NCC1(NC(c2ocnc2-c2ccccc2)=O)CC1 C1(C(=O)NC(c2ncc[nH]2)CO)(COC)CCN(C(c2nc(C)sc2C)=O)C1 Cc1nc(=NCCN2CCOC2=O)[nH]c(=NCC(=O)Nc2ccccn2)[nH]1 c1(C(=O)NC2CCN(C(c3cnc(C)o3)=O)CC2F)ccn2nccc2n1 CN1CCCC(C)(C(=O)NC(Cc2ccco2)C(=O)NCC2CCCNC2=O)C1 O=S(=O)(c1cccnc1N1CCC2(C1)CC2(F)F)NCC(F)CO C(c1cccnc1)=CC(=O)NCCOCCNC(c1cn(CCCC#N)nn1)=O C(CC(C)C)(c1cccnc1)NC(=O)NC(c1nccn1C)CC C(C(CC(=O)O)CC(C)C)NC(C(=O)N(C)Cc1ccc(OC)c(Cl)c1)=O c1(CN(C(c2n(C)nnc2)=O)CCN(C(=O)Cn2nccn2)CC)cccc(Cl)c1 C(=O)(CCCS(C)(=O)=O)N1CCC(C)(CNC(C(C=C)(C)O)=O)CC1 C1(NC(C(C)(C)C2CCN(C(=O)Cc3ccccn3)C2)=O)COCC(C)(C)C1 c1(CC(=O)NCC(CNC(=O)C(C)NC(=O)C2CC2)OC)n[nH]c2c1CCCC2 c1(CC(=O)NC(CSC)C(=O)O)cc(F)c(Cl)cc1Cl C1(NC(C(C)OCCC(C)C)=O)CCC12CN(C(c1cn(C)[nH]c1=N)=O)C2 O=C(CC1=CCOCC1)N1CC(OCCC(=O)N2CC(n3cnnc3)C2)C1 CCCCCC(O)CC(=O)NCC(CC12COC(C1)C2)NC(c1sc(C)cc1Cl)=O C#CCCCC(C)C(=O)NCC(C(C)(C)C)NC(C1CCc2n[nH]cc2C1)=O N1(C(c2cc[n+]([O-])cc2)=O)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C(CO)C1 c1(SCC#C)cccc(C(=O)NCC2CCCN2C(c2ccnc(C)c2)=O)c1 N1(C(CSCCCC)=O)CCC(CO)(CNC(c2nn(C)cc2C)=O)CC1 C1(NC(c2c(C)noc2C)=O)CC(C(F)(F)F)CN(Cc2cc(Br)ccc2I)C1 C#CCC(C)(C(=O)NCCc1nncn1C)NC(c1cc(C)on1)=O CC(C)CCCC(=O)N1CCC(C(C)CNC(=O)CC(O)CN(C)C)CC1 N1(C(c2onc(C)n2)C)CC2CCC1CN2C(c1ccc(O)cc1)=O N1(C(C(C)C(C)O)=O)CCOCC(CNC(c2scnc2Cl)=O)C1 N1(C(=O)CCC2CCCCCC2)CCC2CN(C(C3(O)CCOCC3)=O)CC12 c1(CNC(C2CC(C)(F)C2)=O)nc(CNC(=O)CS(C)(=O)=O)cc(O)n1 CCC(C)(CNC(=O)CC1CN(C(=O)CC2CSCCO2)CCO1)CO C(CC(=O)NC1(CO)CC1(C)C)(C(F)(F)F)NC(CNC(C)=O)=O c1(OC)cc2[nH]cnc2cc1C(N1CCCC(C)(OC)C1)=O C1(C(C)NC(CCn2ncc(C)c2)=O)CCCCN1C(=O)CC(C1CC1)C1CC1 c1(CC)ccc(C(N2CCC(NC(C3CC(F)(CO)C3)=O)CC2)=O)c(N)c1 C1(CN(C(=O)CC2(N3CCCCC3)CCCC2)C)CCCN1C(C1(C)CCC1)=O C(N=c1cc(C)[nH]c(=NCC2CCc3nnc(C)n3C2)[nH]1)C1CC(OC)C1(C)C Cc1ccc(C(N2CCC(CCC(=O)NC3CC4CC(=O)C3O4)C2)=O)c(O)n1 c1(C(=O)Oc2nnc(N(CCOC)C3CC3)o2)ccc(-c2ccco2)[nH]1 Cc1cccc(C)c1CN(C(=O)CNC(=O)CN1CCOC(C)(CN)C1)C N1(C(C(C(CC)O)C)=O)CCC=C(C(=O)NCC2CC(F)(F)C2)C1 CCCCC(O)C(=O)N1CC(CC(C)NC(=O)C(C)C(O)Cc2ccccc2)C1 C1(C(N(c2cn(C)nc2)C(C2CC2)C2CC2)=O)CCC(N2CCOCC2)CC1 c1(CNC(C2C(NC(C3COCC(C)O3)=O)CC2)=O)cccc2ccnn12 c1(C(N2CC(C(C)NC(C3(C)CCCCO3)=O)C2)=O)ccc(O)c(Cl)n1 Cc1cc(-c2cnc(CNC(c3ccc(C(F)(F)F)nc3C)=O)nc2)cc(C)c1 N1(C(c2[nH]cc(C)c2C)=O)CC2CCC(C1)N(C(=O)C(C)O)C2 c1(OC)ccc(S(=O)(=O)N2CC3CN(Cc4nc5ccccn5c4C)C3C2)cn1 c1(N2CC(CC=C)(NC(c3cncc(C)n3)=O)C2)ncnc2c1cnn2C1CC1 N#Cc1cc(C(=O)NC2(C(=O)NCC3CCCCCC3)CCSC2)c[nH]1 Cc1cc(CN2CCC(CNC(c3ccn(C(C)(C)C)n3)=O)C2)no1 c1(NC(C2N(C)CCC2)=O)ccc(Oc2ncc(Br)cn2)cc1.C12CN(C1)C2=O Cc1onc(C(=O)N(C)CCN(C)C(c2ncc(F)cc2F)=O)c1[N+](=O)[O-] N1(C(C2C(C)(CC)C2)=O)CC(NC(=O)CC(CC)C2CC2)CC2(CC2)C1 c1(NC(N(CC(=O)NC2CC2)C)=O)csc(C#N)c1.C12CC1CNC2=O c1(C(=O)NC(CC(=O)NCCOC(CC)(C)C)C2CC2)cc(C)cc(F)c1 CC1=NNC(=O)C1CC(=O)NCC1(F)CCC(CNC(c2ccc(F)cn2)=O)C1 c1(C(N2CC3C(CNC(C4(CC)COC4)=O)C3C2)=O)ccc(F)c(CO)c1 C1(CC)C(NC(=O)CN2CC3CC3C2)CCCN1C(=O)CC1COCC(C)O1 c1(CSC)cc(C(=O)N(CCCNC(C2CC2(C)Br)=O)CCO)sc1C C(=O)(C1=C(Cl)CCC1)N(C1CN(C(C2(n3nccn3)CC2)=O)CC1F)C C(=O)(CC(C)CNC(C1CC(OC)C1)=O)N(C(C#C)C)C CCC(C)C(C(=O)NCC1C2CC1N(C(=O)C1=NOC(C)C1)C2)NC(C)=O C(C(=O)N(C1CC1)CC1CCCN(C(=O)C=CCCC(C)C)C1)(C(C)C)OCC C1(c2nn[nH]n2)(NC(C2CCC3(CC3)CN2)=O)CCC2(CC1)OCCO2 N#Cc1cccc(F)c1C(=O)NC1(CN=c2[nH]cncc2Cl)CCOCC1 N1(C(=O)OC(C)(C)C)CCC(C(=O)NCCc2cn(C(C)(C)C)nn2)CC1 c1(CNC2CCN(C(c3ccn(C)n3)=O)CC2F)cc(F)c(C#N)c(F)c1 c1(C2C(C(N3CC(NC(C4CCC4)=O)C(F)C3)=O)C2)cccc(Cl)c1F CCC(C)C(O)C(=O)NCC1(C(N2CCCC2C#N)=O)CCCCC1 C(=O)(C1=C2CCN=C2NC=C1)N1C2C(NC(c3ccc(O)nn3)=O)C(C2)C1 CC(N=[N+]=[N-])C(=O)NCc1cc[nH]c1C(N1CC(Cc2ccoc2)C1)=O Cc1cnc(C(=O)NC(CNC(c2ccc[nH]2)=O)C(C)C(C)C)c(F)c1 c1(CC(N2CCC(NC(c3cccc(C)c3Cl)=O)C2)=O)ccc2c(c1)COCC2 c1(C(N2CC3=C(C2)CN(C(=O)COC(F)F)C3)=O)cc2cc(F)cc(F)c2o1 N1(C(C2N(C)CCC2)=O)CC(CNC(=O)C=Cc2ccco2)OC2(CCC2)C1 c1(C(N(CC(C)NC(c2ccccc2)=O)C)=O)cncc2cnccc12 N1(C(c2ncc(C)o2)C(=O)NC2CCC2)CCC(C2CCCC2(C)C)C1 C1(CCO)(NCc2c(CC)cco2)CCCCC1 N1(C(C(C=C)O)=O)CCC2(CC1)CN(c1nc(C(F)(F)F)cc(C)n1)CCO2 N1(C(C(C=CC)O)=O)CCN(C(=O)CCCc2nc3ccccc3o2)CC(O)C1 C1(COC)(NC(=O)Cc2cccc(OC)n2)CCCN(C(c2cnc(O)o2)=O)C1 C1(F)(C(=O)NCCC(C)NC(c2cccc(OCC)c2)=O)CCS(=O)(=O)C1 O=C1C(N2CCCNCC2)CCCCN1Cc1cccc(OC(F)(F)F)c1O C12(NC(C3CN(C4CCCCC4)C3)=O)CCCC1CN(C(c1cscc1Cl)=O)C2 Cc1ccc(=NCCC(=O)NCC2CCCCN2C(=O)C(O)C2CCC2)[nH]c1 N1(C(c2ccc(CCC)[nH]2)=O)CCC(C)C(CNC(=O)Cc2c[nH]ccc2=O)C1 O=C(C1=CCN(C(C2CN3CCC2CC3)=O)C1)NCc1ccccc1Cl C1(C(c2ccnc(F)c2)NCC2CCCOC2)(OCC(=O)OC)CCOCC1 C(CCC(C)C)=C(C)Cc1nccs1 [N-]=[N+]=NC1CC(C(=O)NC2CC(CNC(c3ccnn3CCCO)=O)C2)C1 C(=O)(CCS(N)(=O)=O)N(C(CN)C1CC1)C.C1(C(=O)NC)CN2CCN1CC2 CCC(C)(C)CCCC(=O)NC(C)C(C)C(=O)N(C1CN(C)C1)C C1(NC(C#CCNC(C2(C)C(C)OCC2)=O)=O)CC2(C1)CC(C#N)C2 N1(C(CNC(=O)OCC)=O)CCCC(CC)(NC(c2c[nH]c(C)cc2=O)=O)C1 C(=O)(C#CC1CCOCC1)N(CCC1CCN(C(C(CC)F)=O)CC1)C c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC(C)C(NC(=O)CCCCOC)C1)=O c1(SC)ccc(-c2nc(C3CCC(C)C3)n(-c3ccnnc3)n2)nc1 C1(C(N2C(CN(C(C3CC=C(C)CC3)=O)C)CCC2)=O)CCCCCN1C C1(C(=O)NC2CCC(NC(=O)CC3CCC(=O)N3C)C2)(OC)CCCCCC1 N1(C(CC(CC)(F)F)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)CC2)CC1C c1(OC)ncc(NC(C2(C)CCN2C(c2[nH]cnc2C)=O)=O)cc1F C1(C(N2C(CNC(C3(C)CCC3)=O)CCCCC2)=O)C2CC3CC(C2)CC1C3 C1(C(=O)OC)(COC)CCCCN1C(c1cc(F)ccc1C)=O N1(C(CC)=O)CCOC2(CCC(N=c3[nH]c4ccc(Br)cc4s3)C2)C1 C#Cc1ccc(C(=O)NCC(C2CC2)NC(c2sc(C3CC3)nc2C)=O)cc1F c1(C(=O)OC)ccc(Cl)c(C(N2CCC(n3nc(C)cc3C)C2)=O)c1 C=CCCCC(=O)NC1CCCC(CNC(C2(NC(C)=O)CCC2)=O)C1 C=CC(CCC)CC(=O)NC(CCSC)C(=O)NC1CC(=O)N(O)C1 N1(CCCC)CCCCC1C(=O)NC1CC(CNC(c2cc[nH]n2)=O)C1(C)C N1(C(c2c(C)cc(Br)cc2)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1F c1(NC(C2(CC)CNC(=O)C2)=O)ccc(NC(=O)C(C)C(C)(C)C)cc1C S(=O)(=O)(c1cccc2cccnc12)N1C2CN(C(CNC(=O)CCl)=O)CC1CC2 C(=O)(CC(C(F)(F)F)n1cccn1)N(C1CCCN(C(=O)C=CC2CC2)CC1)C N1(C(C(C)OC2CCCC2)=O)CCC(C)(C(=O)N(C2CC3(CCC3)C2)C)C1 c1(C(N2CC(N(C)C(c3cnnc(O)c3)=O)C2)=O)n[nH]c2c1COCC2 c1(C(N2CC(O)(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl N(C)(C1CN(C(=O)C=CSC)CCc2ccccc21)C(C(C1CCC1)OCC)=O N1(C(c2c(CC)c[nH]n2)=O)CCN(C(c2ccccc2C2CC2)=O)CC(C)(C)C1 C1(C(=O)NC2C=CCN(C(c3cc(CSC)c(C)s3)=O)C2)CC2CCC1CC2 N1(C(C=Cc2c(C)nsc2)=O)C2CC1CN(C(c1ccc(CO)o1)=O)C2 C12(NCCNC(=O)Cn3nnc(=O)[nH]3)CCC(CC1n1cc(C3CCC3)nn1)C2 C=C1CCN(C(=O)C(C)C(F)(F)F)C(C(N2CC(Cc3ccoc3)C2)=O)C1 O=[N+]([O-])c1cnc2c(F)cccc2c1N1CCc2cc(C(F)(F)F)ccc2C1 c1(C(C)=O)ccc(C(F)(F)F)c(Cc2cn(CC3COC(=O)O3)nn2)c1 N#Cc1cc(F)c(C(=O)NCCCNC(C2CCc3nncn3CC2)=O)c(F)c1 C(CC(=O)N(C)CCn1cccn1)(C(F)(F)F)NC(CCCCOC)=O CCS(=O)(=O)NNC(=O)c1c(F)cncc1Br C(CN=c1[nH]c(N2CCN3CCCCC3C2)nc2c1COCC2)OC1CN(C)C1 CC1CN(C(c2nccs2)=O)CC(C)N(C(=O)CCN2CCC(O)CC2)C1 C=CCC(C)(CC)C(=O)NC(C1CN(C(c2nnn(C)c2N)=O)C1)C C1(N2CC2=O)CCN(CCC2CCCc3ccccc32)CC1.N1(CC)CCCCC1 c1(CC(=O)NC(C(C)C)CNC(=O)C2=COCC2)ccc2nsnc2c1 C1(CN(C)C(C2CC2Cl)=O)CCN(C(C2CCCN(c3cnccn3)C2)=O)CC1 C(C(O)C(=O)NC(C)(C)C(=O)NCCc1ncn(C)n1)OC C(C(C)(C)C(C)(C)C)CC1C(c2nnnn2C)(NCCCc2cnc(C)s2)COC1 O=C(C#Cc1ccccc1)N1CCCC1C(=O)Nc1cccnc1O C1(OC(C(=O)N(CC(=O)Oc2c(C)ccc(Cl)c2)C(C)C)C)CC(C)(C)OC1(C)C C(=O)(CCCCCC(C)C)NCC1N(C(c2c(C)scc2)=O)CCCC1C CCCCC(C(=O)NCC=CC(N1CCC1C(=O)NC1(CO)CCC1)=O)C(C)C C=CCCC(C)(C)C(=O)N1CCCC(C)(NC(c2cnn(CC=C)c2)=O)C1 CN1CC=CCC1CC(=O)NC1CCCC1CNC(C1(C)CNC(=O)C1)=O c1(C(N2C(C)CN(C)CC2)=O)ccc2c(-c3ccc([N+](=O)[O-])nc3)nn(C)c2c1 N1(C(CCOC2CN(C(C3(C)CC3(F)F)=O)C2)=O)CC2CCC(C1)O2 CC1CC2CN(C(C3(NC(=O)CCC4CC(C)C4)CC(CO)C3)=O)CCN2C1 C1(C(N(C2CCC2O)C)=O)CC(O)CN1C(c1ccc(Cn2ccnc2)cc1)=O c1(CN(C(=O)C(=O)C(C)(C)CC)C(C(CCC)CC)=O)ccc2ncccc2c1 C1(C)(C(=O)NCC(CC2CC2)OC)CC(O)CN1C(c1ccc(F)cc1F)=O N1(C(C(C)OC)=O)CCC2(CC1)CC(C(=O)Nc1cnc(Br)cc1C(N)=O)CO2 N1(C(C(C)CO)=O)CCCC(C)(C)C1CNC(C1(CN(C)C)CCCCC1)=O CC1=C(C(=O)NC2CC(OCC(=O)NC3C4CCCCCC34)C2)CCCO1 C1(CN(C)C(C2(CCO)CC2)=O)CCCN(C(C2(C(C)(F)F)CC2)=O)C1 C(=O)(CC(C)(O)COC)NCC(CC)NC(c1sccc1C(C)=O)=O C1(NC(c2ccccc2)=O)CCCC12CCN(c1nccc(N3CCCC3)n1)C2 C1(C(N(C)CC2(NC(=O)CSC(F)(F)F)CC2)=O)CCOC1=O CCCCC(CC)CC(=O)NC(CC)CCC(=O)NCc1nnc(O)o1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CC2(C1)SCCC2NC(=O)CC1C=CCC1 N1(C(C(COC)O)=O)CCc2c(ccnc2S)C1 c1(CC)cccc(CC)c1CC(=O)NC1CCC1NC(c1ccncc1F)=O c1(OCCNC(CCC)(c2nnnn2CC)C2CC2)ccc(C)c(F)c1 c1(C(N2CC(NC(c3ccc(C)cc3)=O)C(F)C2)=O)n[nH]c2c1COC2 N1(C(CN(CCOC)C)=O)CCC(NC(c2cccc(CO)n2)=O)C2(CCC2)C1 C1(C(=O)NC(C#C)(C)CC)CC2CC2N1C(=O)C(N1CCCCC1)C N1(C(C2(CC)CCNC2=O)=O)CCC2CN(C(=O)C=CBr)CC2C1 c1(C(N2CCC3(CCC3)C2)=O)coc2c1CSC2 N1(C(C(C(C)C)N(C)C)=O)CCN(C)C(CNC(C2(CO)CC2(F)F)=O)C1 C(C(C)(C)CNC(c1cnc[nH]1)=O)N(C(=O)C(F)(Cl)c1ccccc1)C C1(C(N2C3CN(C(C4CC4C(F)(F)F)=O)C(CC3)C2)=O)CCC2(CCCO2)CC1 Cc1ccc(NCc2ccc(C(N)=O)cc2)cc1-c1ccc(CO)nc1 N1(C(C(CC#C)(C)C)=O)CC=C(C(=O)NC2CCCCC2(C)O)CC1 N1(C(CC2C(CNC(COC3(C#C)COC3)=O)C2)=O)C2CCCC1CC2 N1(C(C)=O)CCCN(C(c2c[nH]cc2C2CC2)=O)CC1C C1(N(C)C(c2coc(Br)c2)=O)CCN(C(=O)CCCc2cnn[nH]2)CC1 C1(C)(C(=O)NC2CC(C)(NC(CCCNC(COC)=O)=O)C2)CCN(C)C1=O c1(NC(C)=O)ccc(CNC(C)C(c2ccc(Br)cc2)OC(C)C)cc1 N1(C(C(CO)N(C)C)=O)C2CCC1CC(N(C(=O)Cc1cncnc1)C)C2 Cc1[nH]nc(C(=O)N(CC(=O)NC2C(=O)OCC2CO)C)c1C CC1CCn2ncc(C(=O)NC(c3c(Cl)nc4ccccn34)=O)c2C1 N1(C(c2cnc(C)o2)=O)CCCC(C2CC2NC(C2(C)CCCS2)=O)C1 C1(NC(=O)C=CCOCc2ccccc2)COCCN(C(=O)CC2CC2)C1 c1(CC)cccc(C(N2CC(NC(=O)Cn3cc(CSC)nn3)C2)=O)c1F Cc1cnc(F)c(CNC(C2CC23CC(NC(C2CC2Cl)=O)C3)=O)c1 c1(C2C(C(=O)NC3(COC)CCOC3)CNC2)ccccc1 c1(C(=O)NCCCCCCNC(C2C(C=C)(C(F)(F)F)C2)=O)c(C)nc(C)n1O CC1(C)CCC(C(=O)NC2CCC(NC(=O)CCc3ccc(C(F)F)cc3)C2)O1 c1(OCC(=O)NCC(CO)NC(C(CCC)C)=O)ccc(Cl)c(C)c1 C1(C(=O)NCC(F)CO)COCCN(C(c2ccccc2O)=O)C1 C=CCC(CC=C)C(=O)NCC=CCC(=O)NCC1CC1(Cl)Cl c1(C(c2n(CC=C)nnn2)NCc2ccc(OC)cn2)cccc(C(N)=O)c1 C(=O)(C1=CCC(F)(F)CC1)NCC12CN(C(C(C)C(C)O)=O)C(CC1)C2 c1(C(N2C3CCN(C(CS(N)(=O)=O)=O)C(C3)C2)=O)nncc2c1CCCC2 c1(OC)ccc(NC(C2(F)CN(C(=O)Cn3nc(C)cc3C)C2)=O)c(C)n1 C1(NC(CCN(CC)CC)=O)CN(C(c2cc(C3CCC3)on2)=O)CCC1CO CCC(C)(C)C(=O)C(=O)NN1CCCC1C(=O)NC1CCC2CCC1C2 C(C(=O)NCC1CCCN1C(=O)C(O)CN1CCOCC1)(C(C)C)SC n1(CC)cc([N+](=O)[O-])c(N2CCN(C(c3cc(Cl)c(Cl)s3)=O)CC(O)C2)n1 N1(C(c2cc(C)c(F)nc2)=O)CC(NC(=O)C(C)Cn2ccnc2)CC2(CC2)C1 C(=O)(CC(C)COC)NC(CC)CNC(c1cnc(C(C)=O)s1)=O Cc1cc2c(cc1C)C(C(=O)NC(C)CN(C)C(c1snc(O)c1Cl)=O)CO2 Cc1cc(C)c(C(=O)NCC(F)CNC(c2[nH]c(=N)ccc2C)=O)c(C)n1 C1(CC)CN(C(=O)CCCN(C)C(C)=O)CC1NC(c1cc(C)nn1CC)=O CC(C(=O)NCC1CC(F)CN1C(c1cc(Cl)cnc1O)=O)C(F)(F)F Cc1nc2ccc(COC(=O)C3=CCC(C)CC3)cc2o1 C1(C(N2CCCC2CNC(C2CCOC2)=O)=O)CCCC2CCCCC12 c1(C(=O)NCCCC)ccc(NC(C2CC2Sc2cncc(N(C)C)c2)=O)cc1 C1(C(=O)NCC2(NC(c3cc(OC)no3)=O)CC2)CC2CCCCC2NC1=O O=C(C1=COCC1)NCCSCC=CC(=O)NC1CCCC(O)C1 C(=O)(C(F)C(F)(F)F)N(C1CCN(C(=O)CNS(C)(=O)=O)CC1)C c1(C(=O)NCC2C(COCC)CCC2)ccc(OC)cc1.C12(CC1)C(=O)N2 c1(C(=O)NC2CN(C(C3(CC)CCCC3O)=O)C2)cc(F)cc2nn[nH]c12 c1(-c2[nH]c(=NCc3cccc(COC)n3)sc2)nn(C)c2ccccc12 C1(CC)CN(C(c2ncccc2F)=O)CCC1NC(=O)C(C1CCOCC1)F c1(C(N2CCC(CN(C)C(c3cc(Cl)ccc3N)=O)C2)=O)nc2ncccn2n1 C1(C)(CNC(C2(OC)CCCOC2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)CC1 Cc1cc(C(N2CCCC(c3nc(C)cs3)C2)C(=O)NC(C)C)cc(F)c1 CC1CN(CCCCCNC(c2cc(-c3ccc(F)cc3F)no2)=O)CC(C)O1 C1(C(N(CCN(C(=O)CNC(c2ccco2)=O)C)C)=O)Cc2cccc(F)c2O1 c1(OC)ncc(C)c(CC2(CNC(=O)C(N3CCC(C)CC3)=O)CC2)c1Cl c1(C(=O)NCC2CC(NC(C(CC)NC(N)=O)=O)C2)cncc(OC(C)C)c1 C=CC(C)(O)C(=O)NC1CC(NC(=O)C=CC=CC=CC=CCC)C1 C(CC(C)(C)CC(=O)N1CCC2C(NC(=O)CNC(C3CCOCC3)=O)C12)OC CCCC(CNC(=O)CC1(C)CCN1C(C12CCC(CO1)C2)=O)CCO C1(C(=O)NCc2c(C(=O)NC3CCC(C(C)(C)C)C3)n[nH]c2)C2CCC(F)(F)C12 C(=O)(CCCCCCNC(=O)CNc1cc(C)[nH]n1)N1C(C(CC)O)CCC1 C1(C(=O)N(C)CC2CCCC2NC(C2SCCCS2)=O)(COC)CC1(F)F CC1CN(C2CCN(C(c3ccccc3)=O)C2=O)CC1C(F)(F)F Cc1ccc(F)c(C(N2CSCC2C(N2CC(CC(=O)N(C)CCO)C2)=O)=O)c1 N1(C(C=CSC)=O)CC(NC(=O)CCCC2CCCCC2)CC1(C)C c1(C(=O)NC2CCCC(NC(C3(OC)CC3)=O)CC2)ccc2c(c1)C(=O)CCC2 C(=O)(C(C)(F)CC1CCCC1)NC1C(NC(c2nc(C(C)OC)oc2)=O)CC1 N1(C(C2(CC)CCOC2)=O)CCCC(C2CN(C(C3(F)CCN(C)CC3)=O)C2)C1 N1(C(C(CC)n2ccnc2)=O)CCC(CN(C(=O)CC2(N(C)C)COC2)C)CC1 N1(C(CNC(=O)CS)=O)CC2(CCC1CO)CC2.c1(C2CC2)nc[nH]n1 C#Cc1ccc(CNC(C)(CO)C2CC2)cn1 N1(C(c2ccc(OC)nc2)=O)CC2(CC2)CC1CNC(C1CNC(=O)C1)=O C(=O)(C(CC(F)F)N(C(=O)CC1CCCCN1C)C)NC(COC)C(=O)OC N1(C(C2CCN(C(c3cc(CC)oc3C)=O)CC2C)=O)CCCC2(CC1)CC2 N1(C(CC(c2ccc(C)cc2)(C)C)=O)CC2(CC(NC(C3(CCO)CC3)=O)C2)C1 c1(C(N2CC(NC(C(C)CN(C)C)=O)C(O)C2)=O)ccc2ccncc2c1 N1(C(C(c2cnn[nH]2)N(C(=O)OC(C)(C)C)CO)=O)CCOCC12CCS(=O)(=O)C2 C1(CCNC(CNC(=O)NC)=O)CSCCN1C(=O)Cc1nnc(C)o1 N1(c2n(Cc3c(C)nc(CC)o3)c(C3CC3)nn2)CCC2(CC1)CC2N C(=O)(N1OC2C=CC1CC2)C1C(CC)CN(C2CCCN(c3nccs3)C2)C1 N1(C(CC2C(OCC)COCC2)=O)CC2CCC(C1)N2C(C1CC=CC1)=O C=CCCC(C(=O)N1CCCC(C)(O)C1)NC(=O)Cc1c[nH]nc1C C1(NC2CC3CN(C(=O)OC(C)(C)C)C2C3)CC2(CO)CCCC12 Cn1nc(C(=O)NCCCC2CCCN2C(=O)C=CCO)c2c1CCOC2 c1(C(N2C(C3CCN(C(C(C4CC4)OC)=O)C3)CCC2)=O)ncccc1C c1(C(=O)NCCCC(C)NC(c2c(O)cc(O)cc2O)=O)cc2cccn2cn1 c1(C(N(C2CCN(C(=O)CN(C)C(=O)C3CC3)C2)CCC)=O)cn(C(C)C)cn1 Cc1ccc(C(N2CCCC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)c(C)n1 c1(C(=O)NCCCCNC(c2ncc(N(C)C)nc2)=O)cccc(Cl)c1F CC1CN(C(=O)Cn2ccccc2=O)CC1CNC(c1cnccc1Cl)=O N#CC(C(=O)NCCCC1CCCN1C(c1cc(Br)co1)=O)C1CC1 n1(CCCC)ncc(C(=O)NCC2C3CN(Cc4nc(C)no4)CC23)c1C1CC1 n1(CC(=O)N(C)CCCCCOCCNC(=O)CCc2ncc[nH]2)cnnc1O CCCC(CC=O)C(=O)N(C(C)CNC(c1cn(C)nn1)=O)C C1(C(C)NC(=O)Cn2nnc(=O)[nH]2)CCCCN1C(=O)Cn1cncn1 CCCCCCC(CC)C(=O)N1CCCC1CN(C(=O)C(CC)CC(F)F)CC c1(CC)nc(C(=O)N(C)CC2CCN(C(c3ccoc3C(F)(F)F)=O)C2)c(N)s1 c1(OC(C(=O)N(CC(C)NC(=O)Cn2ccccc2=O)CC)C)ccc(C)cc1C C1(CN(C(C2COCCN2C)=O)CC)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 c1(C(=O)NCC(C(=O)NC2CCOC(C3CC3)C2)OC)cccc[n+]1[O-] N1(C(C=Cc2ccc(CC)o2)=O)CCN(C(C2CCCCS2)=O)CC1C(F)F C=CC1(C(=O)NC(C2CCCO2)CO)CCN(C(=O)Cc2coc(C(C)C)n2)C1 C(=O)(CC(O)C(C)(C)C)NCCNC(CN(C(C=COC)=O)CC(C)O)=O c1(C(N(C(C)CNC(=O)COCCOCCO)CC)=O)cc(C)no1.SC C#CCCC(O)C(=O)N1CC(OC)CC1CCNC(=O)CC1COC(=O)C1 C1(C(=O)NCCCSCCO)CCC2CCC1N2C(C1CC2(CCC2=O)C1)=O C(=O)(C(CC(C)(C)C)NCCSc1ccc(OC)cc1)NCCOC C(CN=c1[nH]c(=NCC2CCCCC2NC(N)=O)c2cc(Cl)ccc2[nH]1)CC N#CC1(C(=O)NCCCCCC(=O)N2CCN(C3CC3)CC2)CCCOC1 C1(O)(C(=O)NC(C2CCCO2)(C)C)CC(F)(F)C1 c1(CC)cccc(C(=O)NCC2COC(CNC(c3ccc(Cl)s3)=O)C2)c1 C#CCCCC(C)(c1nnnn1C(C)C)NCc1cc(C(=O)OC)no1 N1(C(C2CCC(=C)CC2)=O)CC2CCN(C(=O)CC3CC3C3CC3)CC(C2)C1 N1(CCC(C)=O)CCCC(NCc2cc(N3CCCS3(=O)=O)ccc2F)C1C c1(OCC(=O)NCC(CNC(C(C(C)(F)F)Cl)=O)O)ccc2ccccc2c1 C(=O)(C(C)(C)CN(C(=O)CCN(CC)CC)C)N1CCC(CCCC)C1 C12(C(=O)NCC3(C(=O)NCCC4(O)CCOCC4)CCC3)CCCN1CCC2 C1(CCC(=O)N(CCSC)CC)CCCN1C(=O)C(C)O C1(NC(CCc2ccn(C)n2)=O)CS(=O)(=O)N(C)C1(C)C c1(C(N2CC3CN(Cc4c(OC)cccn4)C3C2)=O)ccc(C#N)cc1C N1(C(CC2CC(=O)C2)=O)CCC2(CCCC2NC(C2CCCS2(=O)=O)=O)CC1 C1(C(C)C(=O)NC(c2ccccc2)(C)C)CCN(C(c2cc(Cl)ns2)=O)CC1 C1(N(C(=O)Cn2cnc(=N)[nH]2)C)CCC(NC(=O)COCc2ccon2)CC1 c1(SCC(=O)NC2CC(CNC(C3CCS3(=O)=O)=O)C2)nc2ccccc2s1 C#CCC(O)C(=O)NCC1CCN1C(c1ccc(C(F)(F)F)[nH]1)=O C1(Cl)(C(=O)NC2(C(N(C)C)=O)CC2)CC1C(=O)NCC1CC1 c1(C(N(C2CCN(C(=O)CC3COCCO3)C2)CC)=O)ccc(C)c(F)n1 c1(C(=O)NCC2C3CN(C(=O)CSC45CC(F)(C4)C5)CC32)ccccc1Br c1(C(C(=O)N(CCCNC(=O)C=CCO)C(C)C)O)cccc(Cl)c1 c1(OC)cnc(C(=O)NC2CC(CC(N3CCC3C(N)=O)=O)C2)cn1 c1(-c2nnc(N3C(CCC)CCCC3)n2CC2CCCO2)cc(C)ccc1F c1(OC)ccc(C(N2CC(OC)C(NC(C3(N=[N+]=[N-])CC3)=O)C2)=O)c(Cl)c1 C(=O)(CC(C)C(=O)NC(C(N1CC(C)(N(C)C)C1)=O)C1(C)CC1)OC CC(C)(C)C(C)(C)C(=O)NCCC1CC(NC(=O)C(F)CC2CCOC2)C1 C12(NC(C3CCC4CC4C3)=O)CCCC1N(C(c1cnc3n1CCC3)=O)CCC2 CC1OCCC1NC(=O)CONC(=O)CN1CC2CC2C1 c1(CN2CC3(C(C(N4CCOC(CO)C4)=O)C3)C2)c(O)ccc(F)c1Br N1(C(CCC=CCC=C)=O)CC2CC2(NC(c2cnc(S)nc2)=O)C1 Cc1cccc(CC(N2CCC(N(C)C(C3(C)CCN(C)C3)=O)C2)=O)c1C C1(C(=O)NCCCNC(CC(=O)NCC#C)=O)CCCC(C(=O)OC)C1 C=CCC(C)(C)C(=O)N1CCC(NC(=O)Cn2ncn(C)c2=O)C(C(N)=O)C1 c1(OC)c(C(N2CCC(N3CCN(C)CC3)CC2C)=O)cc(Cl)cc1C C(=O)(C(F)(F)Cc1ccc(F)cc1)NC1CC(CCNC(COCCC=C)=O)C1 C(=O)(C(O)CC(C)(C)C)N1CC(C)C(NC(=O)CCN2CCCS2(=O)=O)CC1 Cc1nc(C2(NC(=O)C(C)N3CCCC3)CC2)no1.C12(CCC1)CC(=O)N2 CC#CCC(C(=O)Nc1cnc(O)c(C)c1)NC(C1CC(C)(C)CCO1)=O C1(NC(CN(C)C2CC2)=O)CC2CCC(C1)N2C(C1CCCC1(C)C)=O C1(CC(C)=O)(C(=O)NC2CC(NC(=O)C(C)NC(C)=O)C2)CCC1 C1(N(C(CCCOC)=O)C)CCCN(C(=O)C(C(C)O)N(C)C)C1 c1(CN2C(C(=O)OC)CC2)c(C)cc(OC)cc1O.C=CCCN1CC1 C(=O)(CC(C)(C)CN(C)C)N1CCC(CNC(C(CC=C)C)=O)(COC)C1 C1(CN(CCCCNC2CCCCC2)C(=O)CC2CCCCC2)CC2CCC2C1 c1(OC)cc(-c2nc(-c3cncnc3)nn2Cc2ccsc2)n(C)n1 O=C(C#CC1CCCOC1)NCC1COCC1NC(=O)C(C1CC1)C1CC1 c1(C(=O)NCC(CNC(C(C(=O)NC)(C)C)=O)CO)cnn2c1N(C)CC2 c1(C(N2CCC(N(C(CCCC(C)=O)=O)C)C2)=O)ccccc1S(C)(=O)=O O=C(C1=Cc2ccccc2OC1)NC1CC(NC(c2cc(F)cc(F)c2)=O)C1 CCC(C)(C)C(=O)N1CC(CNC(c2cncnc2-c2ccccc2)=O)C(O)C1 CC(C)C(C(=O)N1C(CNC(c2cccn2C)=O)CC2CC12)c1ccc(F)cc1 c1(CC)ccc(O)c(NC(=O)CC(CC)NC(c2cc(C(N)=O)[nH]n2)=O)c1 C1(CC(=O)NCC(=O)N(C2CN(C)C2)C)CCCN1C(C1CC1F)=O CCC(O)C(F)(F)C(=O)NCC1CN(C(=O)CC2CCC3CC23)C1 C1(C(=O)NC2CCC(NC(c3ocnc3C3CCC3)=O)CC2)CC2COCC2C1 CCCC(C)(C)C(=O)N1CCCC(CO)C1.N12CCN(CC1)C(=O)CCOCC2 c1(CCC(=O)NCC2(F)CC(CNC(=O)CCC3CC3)C2)ccc(Cl)c(F)c1 C(CCCCCC(=O)N(C1CCCC1)CC)NC(c1c(CC)ncs1)=O C(=O)(C(O)(C(F)(F)F)c1ccccc1)NC(CNC(=O)C(F)C1CC1)C1CC1 n1(CC(N2CC(N(C(=O)C3=CCOCC3)C)C(F)C2)=O)ncn2nccc2c1=O C(c1cccc(F)c1Cl)=CC(=O)NC1C(NC(C=CC=CC)=O)CCOC1 CC1(NC(C23CC(F)(C2)C3)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 n1(C(CC)C)nc(C(=O)NCC(CNC(=O)Cc2ccsc2)CO)cc1C C(C)(C(=O)N1CCC(CNC(c2cccc(N)n2)=O)C(O)C1)(C(C)C)NC(C)=O C1(C(=O)N(C)CCn2cncn2)CC(NC(C(=O)NC)=O)C12CCC2 c1(CC)ccccc1Cl.C12CCN(CC1)C(c1ccc(C(C)OC)cc1)C(=O)N2 c1(C(=O)NCC(C)(C)CNC(c2cncnc2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CC(=O)NCCNC(Cn2cc(N)nn2)=O)c(F)cccc1C#N.CNC n1(CC)cc(Cl)c(C(=O)NC2CCN(C(=O)CC3CCCC3)C2)n1 Cc1cc(=O)n(C)nc1C(=O)NCCNC(c1cccc(Br)c1F)=O c1(N(CC(C2CC2)OC)C)nc(NC2CCOC2)c2cnn(C)c2n1 C(=O)(CCC(C)(C)C(=O)c1ccccc1)N(CC(=O)OC)Cc1ccc(Cl)c(F)c1 C1(NC(C(CC)OCC)=O)CC2CC(NC(c3cccnn3)=O)CC12 C=C1CCN(C(c2cnn(CCNC(c3ncoc3C)=O)c2)=O)C1 C(=O)(N1OC2CCC1C2)C1(NC(Cc2c(C)ccnc2)=O)CCCCC1 Cc1ncc(C(N2CCOC(CNC(C3C4CNC(=O)C34)=O)C2)=O)c(=N)[nH]1 c1(CC)ncccc1SC.c12cc(n[nH]1)C(=O)NCCOC1CN(C1)C2=O N1(C(c2c(C)cc(CC)o2)=O)CCCC(C)(C(=O)N(C(C)CC2CCOC2)CC)C1 c1(C(=O)NC2C(C)(C)CN(C(=O)CCC[N+](=O)[O-])C2)nc2ccc(Cl)nn2n1 c1(CC)cc(NC(=O)CC(C)NC(=O)CCCCCn2cnnn2)cc(O)c1 c1(N(CCCNC(C2C(CC)OCC2)=O)CC)nccc(S(C)(=O)=O)n1 C1(CC)CCN(C(c2nccn2C)=O)C1C(=O)NCC1CCCN1C c1(OC)ccc2n[nH]c(SC)c2c1.c12cn(nn1)-n1ccc(n1)C(=O)N1CCC21 c1(C(C(C)NC(C(C)=CC)=O)NC(=O)COCC(=O)NCC)ccccc1 C1(NC(CCOCC#C)=O)CCCN(C(c2ccc(OC)c(Br)c2)=O)CC1 C1(NC(C2(CNC(CC=C=C)=O)CC2)=O)CC2(C1)CC21CCC1 c1(CN2CC(CC(=O)Nc3c(O)ccc(C)n3)C2)cc2ncccc2o1 C1(CNC(C(C)(C)OC(C)C)=O)C(C)CCN1C(=O)CCC1OCCO1 C(=O)(C(CNC(C1OCCCC1(C)C)=O)C(C)(C)C)N1CC[Si](C)(C)C1 C1(C(=O)N(c2cn(C)nc2)C2CC2)CN(C(=O)COCC2CCC2)C2(CCC2)C1 CC1CC(NC(C2CC(O)C2)=O)CCN1C(c1cccc(C(F)F)c1Cl)=O c1(C(=O)CN2CCCC2Cc2ccccc2)ncc(C2CCOC2)s1 C(=O)(CCCCC(C)C)NC(CC=C)CC(=O)NCCc1cnco1 C1(C(N2C(C)(CNC(c3ncc(C(F)F)s3)=O)CCC2)=O)Cc2cccnc2C1 C=CCCC(=O)NC(C1CC=CCC1)C(=O)NC(c1nc[nH]n1)C1CC1 C1(C(C(=O)NC2CC(F)(CNC(C3(c4ccno4)CC3)=O)C2)F)CCCCCC1 N1(C(C2C(C)(C)C2)=O)CCC(C2CCCN(C(c3cncc(C(F)F)c3)=O)C2)C1 c1(C(=O)OC)ccc(NC(=O)CCc2cc(C)ccc2C)cc1OCC c1(CC(=O)NCC2C(NC(C(C)c3ccco3)=O)CC2)sc(O)nc1O C1(CC=C)(NC(C2COCCC2(F)F)=O)CCCN(C(=O)CC(C)(C)CC)C1 N#Cc1ccccc1C(=O)NCC(CC(=O)N1CCCC1C(N)=O)C1CCC1 CCC(C)CCCCC(=O)NC1CCCCN(C(C2(CC3CC3)CCCO2)=O)C1 C1(O)(CNC(C(F)=C(C)C)=O)CC(NC(=O)C(O)c2cnc[nH]2)C1 c1(C(N2CCC(C(C)(C)C)(CNC(C(CSC)C)=O)C2)=O)cc(C)c(CO)cn1 c1(C(C(N2CC(N(C(c3c(C)n[nH]c3)=O)C)C2)=O)C)cc(Br)ccc1F C1(C)(COC)CN(C(=O)C(C)(C)C2CCN(C(=O)CCCCN(C)C)C2)C1 C1(C(=O)NCC2(COC)CN(C(=O)Cc3ccsn3)C2)CCCC(=O)C1 c1(OCCC(=O)N(C(C)CNC(C2CC3CC2C3)=O)C)ccc(S(C)(=O)=O)cc1 C(=O)(C(C)C(C)COC)N(CCCNc1ccc(NC(CCC)=O)cc1)CCC N1(C(C2(OC)CCCC2)=O)CCC(NC(=O)Cn2nnnc2C)CC(C)(C)C1 C1(CNC(c2ncc(Cn3cc(COCCCO)nn3)s2)=O)CCCCC1(F)F c1(C(C)NCc2ccc(C(=O)NC)o2)cc2ccccc2[nH]1 n1(CC)cc2ccc(C(=O)NC(C)C(C(C)C)NC(c3c[nH]cc3C)=O)cc2n1 c1(Nc2cccc(SC)c2)ncnc(NC(C)C(C)Oc2ccccc2F)c1C c1(CC)nc(C)c(C(=O)NCC2(F)CCC(CNC(c3n[nH]cc3CC)=O)C2)s1 C(CCCC(=O)NCC1C=CCN1C(=O)CC1CC1c1ccccc1)OCC C(=O)(C1=C(Cl)CCCC1)NCc1ccc(C(N2CCC(N(C)CC)CC2)=O)s1 Cc1ccccc1SCC(=O)NCC1CC2CC2N1C(=O)Cc1sc(O)nc1O c1(CC)nc(C)c(C(=O)NCC2COC(CNC(C3CC(=C4CC4)C3)=O)C2)s1 CCCC(CCCNC(c1sccc1C(C)C)=O)NC(=O)C(C)C(F)F N1(C(CCCN(C)CC2CCCO2)=O)CCC(NC(C2CCC=CCC2)=O)CC1 c1(C(=O)NCC(C(=O)NCCC(C)C)OC)cccc2c1OCO2 Cc1nnc2n1CCCC2C(=O)NC1CCN(C(=O)CCCC#N)CC1 N1(C(c2ccoc2Cl)=O)CCC2CCCN(C(=O)COCC(F)(F)F)C2C1 N1(C(=O)CC2CC2)CC2C3CCC(C2C1)N(C(=O)CC(=O)NC1CCOC1)C3 c1(NC(CC2CC(NC(C3C(C)CC3)=O)C2)=O)ccc(N2CCOCC2)cc1 C=CC1(C(=O)NCC[Si](C)(C)C)CCN(C(C2CCS2(=O)=O)=O)C1 N1(C(CCC=C)=O)CC(NC(=O)C(C)(O)C(C)c2ccccc2)CC2(CC2)C1 c1(CCCC(=O)N(C(CNC(CC(CC)C)=O)C2CC2)C)nc2ccccc2o1 C1(CCC=C)(C(=O)NC(c2ncnn2CC)C)CN(C(c2ccc(OC)o2)=O)C1 C#Cc1ccc(OC)c(C(N2CCC(NC(=O)CC3CC3C(F)(F)F)C2C)=O)c1 C(C(C)C)(C(O)C(=O)NCC1CCN(C(C2CC3(CCC3O)C2)=O)C1)OC C1(C(=O)NCC2(O)CCN(C(Cc3cc(C)no3)=O)CC2)Cc2cccnc2C1 Cc1nc2cncc(C(N3CC(CO)CC3CO)=O)c2[nH]1 C(=O)(CCC(C)(C)F)NC(CN(C)C)C(N1CCCCC1CCCO)=O c1(NC(C2N(C(CCC#C)=O)CCCC2)=O)cccc(C#N)c1 N(C1CCCc2nn(C)cc21)C(N)=O.C1(OC)CC2CC1NC(=O)NC2 C12(NC(c3c(C)nns3)=O)CCCC1(F)CN(C(=O)C(F)(F)C(F)(F)C(F)F)C2 c1(C(=O)NCC2C(CNC(c3cn(C)nn3)=O)C2)cncc(C(N)=O)c1 C1(CC#C)(OC(C2CC(O)CN2C(C(=O)NCC)C(C)SC)=O)CCCCC1 C1(NC(c2c(CC)scn2)=O)CS(=O)(=O)CC1NC(=O)CCCn1cc(C)cn1 C1(C(N(c2ccccc2I)C(C)C)=O)CC(=O)N(CC(F)(F)F)C1 C1(CNC(c2n[nH]c(C)c2C(F)(F)F)=O)CC(N=c2ccc(C#N)c[nH]2)C1 N1(C(CC2N(C(CC3CCC(C)CO3)=O)CCOC2)=O)CC2CN(C)CC2C1 C(=O)(C1CCc2ccccc21)OCC(=O)NCC(COC1CCCOC1)N(C)C Cc1cc(C(C)C(=O)NCC2COCCN2C(=O)CCN(C)CCO)cc(C)c1 c1(NC(C)(C)C)ccc2c(c1)CC(C(N)=O)O2.c12cc(nc(=O)[nH]1)NO2 C(=O)(C1CCCc2nncn21)NC1CC(N(C(C=Cc2c(C)coc2C)=O)C)C1 c1(C(=O)NCC2N(C(COc3c(F)ccc(C)c3)=O)CC2)cnc2[nH]nnc2c1 C1(C(N2CC(C(N)=O)C2)=O)COCCN1C(=O)Cc1cncnc1 c1(CN(C)C(C2CNCCOC2)=O)cc(Br)cc(F)c1O C(=O)(CCCC(C)(C)C)N1C(CN(C(c2nc(O)nc(O)c2F)=O)CC)CCC1 C(C1=CCCN(C(=O)C(C)N(C)C)C1)NC(C(Cc1c(OC)cccc1)(C)C)=O C1(C(=O)NCc2ncn(CCCC)c2)CCNC(=O)C1 c1(N2CCCC(OC)(CO)C2)nc(C)cc(=NCc2c(Cl)cccc2Cl)[nH]1 C1(NC(Cc2c(C)cc(F)cc2)=O)C2COCC1CN(C(C1(C#N)CCC1)=O)C2 CC1(C)CCN(C(=O)CC2CCC2)C(C(=O)NC2(C)CCC(=O)NC2=O)C1 c1(C(C)C)nc(NCCC(O)C2CCCC2)cc(=NCC2CC(F)(CO)C2)[nH]1 c1(N2CCC(C)C(NC(=O)CCC(N)=O)C2)nccc(S(C)(=O)=O)n1 N1(C(CN(CC)CC)=O)CCC(CNC(=O)C=CC2CCCN2C)CC1.C(C)(=O)O N1(C(CNC(c2cccs2)=O)=O)CC(CNC(C2CC3CCC2O3)=O)C(O)C1 c1(CC(=O)NC2CC(F)(CNC(=O)CCC3CCCO3)C2)ccc(O)cc1 c1(CCC)ccc(C(c2cnn(-c3ccc(OCN)cc3)c2)OC)cc1 CCC(F)(F)C(C)(C)C(=O)NCC1(C2CC2)CCN(C(C2CCCC2C)=O)C1 C1(CNC(c2cc(C)nc(C)c2)=O)CC2COCC2N1C(c1onc(C)c1C)=O C(C(=O)NC(CO)CCC1CC1)(C(C)(C)O)NC(CCSCCCC)=O C=C(C)C(C)(O)C(=O)NC1CC(O)(CNC(c2nn[nH]c2Cl)=O)C1 c1(C(=O)NCC(C)CN(C(=O)CC2CC2(C)C)C)csc2cc(Cl)cnc12 c1(CC)ccc(CNC(=O)C(Cn2cncn2)NC(=O)OC(C)(C)C)o1 N1(C(CC(C)N(C(c2c(CC)cncc2)=O)C)=O)CCC(C)(C2CC2)C1 N1(C(CCOc2c(OC)cccc2)=O)CCN(C(=O)CCOC(C)C)CC2(CC2)C1 Cc1nn(CC(=O)NCC(=O)NC(CO)C(=O)O)c(C)c1C c1(CC)cc(C(F)(F)F)ccc1C(=O)NCC(CNC(=O)C(C)C#N)CO CC(C)(CC(=O)NC1CCCN(C(=O)COc2ccccc2)CC1F)CC(F)F c1(NC)c(C(=O)NC2(C)CN(C(C3CCCS3)=O)C2)cccc1[N+](=O)[O-] c1(C(N(C)CC2CCN(C(C(C(C)(C)C)OC)=O)C2)=O)cnc2ccncc2c1 Cc1cc(CN2CCN(C3CCC(N)C3)CC2)ccc1Cl C(=O)(CC1=CCCCC1)N1CCCC(NC(C2CC(=O)N(C3CCCC3)C2)=O)C1 C12(C(N3CC4C(CN(c5cc(C)on5)C)C4C3)=O)CC3CC(C(=O)N1)C2C3 C(=O)(CC1COc2cc(O)ccc21)N1CC(CCNC(c2c(CC)[nH]cc2)=O)C1 C#CCC(C)(C)C(=O)NCCC(C(C)C)NC(=O)CC(=O)OC Cc1nc2ccc(C(=O)NCC(C)(C)CNC(=O)CC3C(C)C3(F)F)cn2n1 c1(OC)cnc(C(N2CCC3C(NC(=O)CCC(=O)N(C)C)C23)=O)c(F)c1 Cc1ncc2n1CCC(C(=O)NCC(O)CCNC(=O)CC(C)(C)C(F)(F)F)C2 c1(C(N(C)CC2CCCN2C(=O)C=Cc2ccccc2Cl)=O)ccc(C#N)c(O)c1 C(N=c1ccnc(C)[nH]1)C1OCCCN(C(CC(CC)(F)F)=O)C1.CC=O C1(NC(C(C)OC)=O)CN(C(c2ccc(Cl)c(N)c2)=O)CCC1CO C(=O)(C(O)CO)NCCCNC(C1(CSC(CCC)C)CC1)=O.c1(S)ccccc1 C(c1c(Cl)nc2ccccn12)=CC(N1CCC(CNC(c2c(C)ncs2)=O)C1)=O N1(C(c2nc(OCC)oc2)=O)CCOC(CCCNC(=O)CS(=O)(=O)NC)C1.CO Cc1cnc(F)cc1C(=O)NC1CCC(NC(=O)C(C(C)C)OCC(C)C)CC1 C(=O)(CCCCC(F)F)N1CC(NC(C=Cc2nnn(C)n2)=O)C(O)C1 C1(C(N2CC(COC)(CNC(c3n[nH]cc3C)=O)C2)=O)CN2CC3CC2(CO1)C3 C1(C(N2CCSCCC2C)=O)(CC)CCCN(C(c2ccc(CC)[nH]2)=O)C1 C1(C(N(CCNC(=O)Cc2cc(O)nnc2O)CC)=O)CCc2nn[nH]c2C1 C1(C(=O)NC(CC)CNC(c2ncc(C)cn2)=O)CC2(CCCC2)C1 C1(C(=O)NC(CNC(c2cc(C(=O)OC)ncc2)=O)C2CC2)CC2CCC(C1)C2 c1(OC)ncc(C(=O)NC2COCC2CNC(=O)Cn2ncn(C)c2=O)c(C)n1 CCC(CC(F)F)C(=O)NCC1CCN(C(c2cc(C(N)=O)cc(C)c2)=O)CC1 C1(NC(c2c(CCC)occ2)=O)CN(C(C2(C)CC2c2ccccc2)=O)CC1O c12ccc(cc1)C(=O)NCC(C)N(C)C(=O)CN2C.c1(SC)ccoc1C1CC1 c1(OC)ccc(C(N2CCCC2(C)C(=O)Nc2c(Br)ccnc2Cl)=O)c(Br)c1 C1(CC(=O)OC)CCOCC1Nc1ccc(-c2cncc(N)c2)nc1 C1(C)(CNC(CC(C)C2CCCO2)=O)CCCN(c2ncnc(O)c2Br)C1 c1(OC)ccc2cc(C(=O)NCC3CCCC3NC(c3ccc(C)cn3)=O)sc2c1 C12(C(N(C3CCN(Cc4onc(CCC)n4)CC3)C)=O)CCCC(C1)OC2 C1(C(N(CCCN(C(C(C2CCC2)OCC)=O)C)C)=O)CCCC2(CCC2)O1 C1(C)(NC(C(=O)N(CCN(C)C2CC2)C)=O)CN(C2CC2)C(=O)O1 C(CC(C)C(=O)NCC1CC(NC(=O)C(=O)NC2CC(=O)N(C)C2)C1)=CC c1(C(C)C)nc(Cl)cc(=NCC23CC(NC(c4nsnc4O)=O)(C2)C(C)O3)[nH]1 N1(CC(=O)N(CC)CC2CCCN2C(=O)C(=Cc2ccco2)C)CCC(C)CC1 C1(C(=O)NCCCN(C(C(Br)=C(C)C)=O)C2CC2)CCN(C2CC2)C1=O C12(C(=O)NCC(C)CN3CCCC3)CC1CN(C(c1sccc1CO)=O)C2 C12(NC(C(C)N(C(C)=O)C)=O)CCC(C1)N(C(=O)Cc1ccco1)C2 CC1CCN(C(=O)CN(C(=O)CC2(CO)CCC2)CC2CC2)C1 C(N=c1[nH]c2c(c(=NCC3(SC)CCOC3)[nH]1)CCC2)c1cc(OC)no1 C(=O)(C(C)(C)COCC(F)F)NC(C)C(C)NC(c1ccncc1F)=O N1(C(C(c2ccc(C)cc2)C)=O)CCC(C2(NC(c3cn[nH]c3)=O)CCC2)CC1 N1(C(CC(CC)c2ccccc2)=O)CCN(C(c2ccc(C)nc2C)=O)C(CO)C1 c1(OC)ccc2c(C(=O)NC(C)CCN(C)C(C3CC(F)(F)C3)=O)cnn2c1 C1(C(=O)NCC2C(C)CCN(C(CNC(=O)OC)=O)C2)CCc2c(cnn2C)C1 N1(C(C2CCC(NC(c3nccc(C#C)c3)=O)C2)=O)CC2CCC(O)CC2C1 C1(C(N2CCN(CCCNC(C34CC(CO3)C4)=O)CC2)=O)CCOC2(CCC2)C1 C1(C(N(C(C)C)CC2CCN(C(CSCCCC)=O)C2)=O)CCC(C(N)=O)N1C C(=O)(C(O)C(F)(F)F)N1CC(NC(=O)CCCCC2CCCCC2)C1 N1(C(C2C(C)OCC2)=O)CC2CCN(C(=O)CCCn3ccnc3)C2C1 Cc1cc(C(F)(F)F)cc(C(=O)NC(C)CC(C)NC(=O)C=CC2(C)COC2)n1 C1(CC(=O)NCC2CCCN(C(=O)COc3cnn(C)c3)C2)(OC)CCCCC1 C(=O)(C(CC(N)=O)NC(=O)CCN1CCOC1=O)NC1CCN(C(C)=O)C1 c1(C(=O)NCC(C)C(F)C(=O)N(C)Cc2cocn2)cncc2[nH]ccc12 c1(C(=O)NC(C)CCNC(c2ccc3c(c2)COC3)=O)ccc2c(c1)C(C)CO2 N1(C(C2(CC)CCCN2C(=O)CCc2cnn(C)c2)=O)CC2CC1C1CC21 N1(C(c2cccc(C)c2F)=O)CCCC(C2CN(C(=O)C=CI)C2)C1 CC1CCN(c2ccc(CN(C3CCCCC3NCCO)C)cc2)CC1 c1(CC(C)C)ccccc1C(N1CC(NC(C2CC2[N+](=O)[O-])=O)C(C(F)F)C1)=O C=C(C)c1cccc(CNC(=O)N(C2COCC2CC)CCN2CCOCC2)c1 c1(CC)nc(C)c(C(=O)N(C)CCNC(c2cc(C(=O)OC)no2)=O)s1 c1(C(=O)NC2C(C)CN(C(=O)C=Cc3cscn3)C2)c[nH]c2ncccc12 C12(C)CCCN1C(=O)CNC(=O)NC2.c12cncc(c1)OC2.C(CC(C)C)SCC CCCC(O)(CSCCc1cccc(CCOC)c1)CCC C(=O)(C(C)C(C)(C)C)NCC(CC(C)C)NC(=O)CCc1ccncc1Br c1(CCC(=O)N(CC(CC)NC(C2CCC(=O)O2)=O)C)cncc(F)c1 CS(=N)(=O)C1CN(C(=O)C=C(C2CC2)C2CC2)C2(CCC2)C1 c1(-c2nc(C(c3cn(CCCCC)nc3C)O)on2)cccc2cccnc12 C(=O)(C1=C(C)N(C)c2ncnn2C1)NC1CCN(C(c2c(OCC)c[nH]c2)=O)C1 N1(C(CCSC)=O)CCC(C2CCN(C(c3cncc([N+](=O)[O-])c3)=O)C2)C1 C(C(C)(C(=O)N(CC(=O)N(C1CCCCC1)C)C1CCC1)OC)OC C(CCO)(C(=O)N1CCOC(CNC(=O)C=Cc2cocn2)C1)N(C)C C1(C(=O)NCCCCN(CCCSC)C)COCCC1(F)F.C1(C)(C=O)CCCCC1 Cc1nc2ccccc2n1CC(=O)N(CCCNC(C1CCCC1C)=O)C(C)C N1(C(=O)COCCO)CCCC(Cc2cn(C3CCN(CC=CBr)CC3)nn2)C1 C(=O)(C1CCCn2nccc21)NC(CCCNC(C1N(CC)C(=O)CC1)=O)(C)C N1(C(CN(CC=C)C2CC2)=O)CCC2(C1)OCc1ccccc12 C1(CC(=O)Nc2cccc(CO)c2)CN(Cc2ccccc2C(F)(F)F)CCO1 CCCC(CNC(=O)Cn1nc(C)cc1C)C(=O)NCC1(C2CC2)CCC1 C1(C(N2C(CN(C(=O)C(F)(F)C3(O)CCCC3)C)CCC2)=O)CC12CCOC2 N1(C(C=CCC)=O)CCC(C(N2CCC(CC)(CN(C)C)C2)=O)C12CC2 C(C)(CC(=O)NC1CC1CNC(=O)COCC1CC1)NC(=O)NC c1(CC)nc(C)[nH]c1C(=O)NCC(C)(C1CC1)NC(c1cnc(C)nc1)=O c1(NC(C2C(NC(CCN(C)C3CC3)=O)CC=CC2)=O)ccc2nccn2c1 CC(C)C(F)(CNC(C1CCCCCC1)=O)C(=O)NC1CCOC2(CCC2)C1 c1(C(=O)NCC(=O)NC2(CNC(CCC(=C)C)=O)CCOCC2)cccc(C#N)c1 C1(COC)CCN(C(=O)C(C2CCCC2)NC(c2cccnc2S)=O)CC1 C1(NC(C(c2c(Cl)cccc2Cl)C)=O)CCN(C(=O)CCF)C12CCC2 Cc1cc(N)n(CC(N2CC(CNC(c3sccc3C)=O)C(C)C2)=O)n1 C1(CC)CCN(C(c2cc(C(C)C)oc2C)=O)C1CNC(C1CCCC(C)O1)=O C12(CC=CCC1)C(=O)NC2.c1(CNC(C2(C)CC(CO)C2)=O)ccc(O)nc1 N1(CCCC)C(=O)CCN(CC(C)(C)F)C1=O C(c1ccccc1F)=CCC(=O)NC(CC)CN(C)C(c1ccco1)=O c1(OCC(=O)NC)cccc(CC(N2CC(NC(C3SCCC3C)=O)C2)=O)c1 N1(C(C(c2ccc(C)s2)C)=O)CCC2(CCC(NC(=O)CCC3CCC3)C2)CC1 C1(CC(=O)NCc2cc(O)cc(F)c2)CCC(F)(F)C(=O)N1 C1(=O)C(F)=CC(=O)N(C)C(C2CC2)CN1.C(CCC=CC)=C(C)C.C(C1CC1)=C C1(N(C)C(c2ccc(CO)s2)=O)CN(C(=O)C(F)CC2CCCCC2)CC1F CP(C)(=O)c1ccc(C(N2CCC2CNC(c2nsc3ccccc23)=O)=O)cc1 N1(C(C2CC2C2CCCCC2)=O)CCC2(CC1)CN(CCOc1ccccc1)C2 C#Cc1cnc(C(N2CC(N3CCN(C(C4(C(=O)OC)CC4)=O)CC3)C2)=O)cn1 C12(CNC(c3ccc(OCCC)cc3)=O)CCCC1CC(=O)N2 C(c1ccc(C)cn1)=CC(=O)NC1C(NC(C(CCC)C)=O)C1 N1(CC(c2ccc(Cl)cc2)C)CC2(CN(C(C3CC3C(C)O)=O)CCO2)C1 C1(CC(N2C(C(=O)OCC)CSC2)=O)CCC12CCNCC2 c1(C(=O)NCCC(C)OC)cccc(CNC(=O)Cc2cn[nH]c2)n1 C1(C(=O)NC(CCOC)CO)CCCN(C(c2cnc(O)c(C)c2)=O)C1C C1(CCNC(=O)CSCC2CCCO2)CN(C(c2cnccc2Cl)=O)CCCO1 C(CC(C)C(=O)N1CCN(C(=O)CN(C(=O)C(C)(C)C2(O)CCC2)C)CC1)OC c1(C(CC)C(=O)NCCCNC(=O)C=C2CCC(C)C2)c(C)noc1C c1(C(N2C3C(NC(Cn4nnc(C)n4)=O)CC(C3)C2)=O)ccsc1S(C)(=O)=O c1(NC(c2cc(-c3ncsc3Cl)ccc2F)=O)c(F)cc(F)cc1Br C1(CC)CCN(C(C2CC2[N+](=O)[O-])=O)C1CNC(=O)CCn1ccnc1 c1(C(=O)NC2(CNC(C(C)=CC)=O)CCOC2)cn(C)c(=O)nc1O c1(OC)ccc(CC(N2CC3CC3(C(=O)NC3CC3(C)C(F)F)C2)=O)cn1 C1(C(=O)NCC(c2cnn(C)c2)C)C2CN(CC3(c4ccc(O)nc4)CC3)CC12 c1(C(N2C(C(N3C(CC)CN(CC)CC3)=O)C=CC2)=O)cccc2c[nH]nc12 c1(C(N2C(C(CNC(C(CC(C)C)C)=O)(C)C)CCC2)=O)cccc2c1NCC2 C(=O)(C=C(Cl)Cl)NC1(CNC(C(C)SCCCC)=O)CC1 Cc1ccc2c(CC(N3CC(CNC(C4CC(F)(F)C4)=O)C(C)C3)=O)c[nH]c2c1 C(c1ccccc1F)=CCNC(C(C)(C)C1CCN1C(C1CCCS1(=O)=O)=O)=O N1(C(C2(OC)CCCC2)=O)CC(NC(=O)CN2C(=O)CCC2=O)CC(O)C1 N1(C(C(C)OCCOC)=O)CCN(C(C2(C(C)C)CCOCC2)=O)CC12CCC2 N1(C(C(=O)NCC2C(C)(C)C(F)(F)C2)=O)CCC12CC(C)(CO)C2 C1(C(=O)NCC2N(C(Cn3ncc(CC)c3)=O)CCC2)C2CCCCCCC12 C12(C(=O)NC3CCC(NC(CN(CC)CC)=O)CC3)CCCCC1CS(=O)(=O)C2 c1(CC(=O)NCc2nc(C(N3CCC3C3CCCCO3)=O)co2)ccc(Cl)cn1 C(=O)(C(C)(O)C(F)(F)F)NCCCCN(C(c1c(C)cnnc1)=O)C c1(C(=O)NC2C(NC(=O)CN3CCOC3=O)CC2)ccn2nnnc2c1 Cc1cc(NC(=O)Cn2cnnn2)ccc1NC(=O)Cn1cncn1 CC(C)C(C(=O)NCCCCn1cc(C2CCCCC2O)nn1)c1ccn(C)n1 CS(=O)C1CN(C(c2cc(CNC(C3CCCCC3)=O)no2)=O)C1 CCCCC(C(=O)NC(C1CCCCC1)C(=O)NCCC(C)C(C)(C)C)N(C)C CC1C(C)N(C(=O)Cc2ccco2)CCN1C(=O)CCc1nnc(C2CC2)o1 c1(CN(C(=O)C(=O)N(C)CC2CC3CCC2C3)CC=C)ccc(F)cc1 c1(C(N(CC(C)CNC(C2CC23CC(F)(F)C3)=O)C)=O)cccc2[nH]ncc12 C1(C(=O)NCCC(=O)NCC)CCCC(CNC(=O)COc2ccncc2)C1 N1(C(CSCCC#N)=O)CC2CCC1CN(C(=O)CN1CCCC1=O)C2 N1(C(CC2(C)CCCO2)=O)CCCC12CCN(C(c1csc(F)c1)=O)CC2 CC1COC(C(=O)NC(C)(C)CN(C)C(c2csc(C(N)=O)n2)=O)C1 Cc1nn2ncccc2c1C(=O)NC1CC1CNC(=O)CCOCC(F)(F)F Cc1ncc(C(=O)NCC2CCC(NC(C3CC4CC4C3)=O)C2)o1 c1(C(N2CC(O)CC2CNC(C2(CC(F)F)CCC2)=O)=O)cn2ncccc2n1 c1(C(=O)NCC(C)CN(C)C(c2nn(C)cc2[N+](=O)[O-])=O)nc2ccccc2[nH]1 c1(C(C)NC23CCCC2CN(C(=O)C(C)(C)CO)C3)ccc2c(c1)CCCC2 N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(=O)CC2CNC(=O)C2)CC12CCC2 C(C(C(=O)NCc1ccc(C)c(C)c1)C(C)C)NC(CCCN(C)CC)=O N1(C(CNC=O)=O)C2CC1CN(C(=O)CCCC1OCCO1)C2 c1(C(=O)NC2(C(=O)NCc3cncc(O)c3)CCOCC2)cc2ccccn2c1 c1(C(=O)NC(CNC(C#CC(C)(C)C)=O)CO)c[nH]ccc1=Nc1ccccc1 Cc1cc(Cl)c(CN2C(C(=O)Nc3cnc4ncnn4c3)CCC2C)c(Cl)c1 CC(C(=O)N1CC(NC(C2CC(F)(CO)C2)=O)C(F)C1)C(C)(F)F N1(C(C=CCOC)=O)CCN(C(=O)C(c2cc(Cl)cc(Cl)c2)O)CC1CF C(C(F)(F)F)(C(F)(F)F)c1n(Cc2ncc(Cn3ncc(C)c3)cn2)nnn1 C1(C(N2CCCC(CCF)C2)=O)CC(F)(F)CN1C(C1CCOC1)=O c1(N2CC(CN(C(=O)C=Cc3ccccc3Br)C)C2)cc2ncnn2cn1 CCC(CC(=O)OC(C(=O)NOCCOC(C)C)C1CCCO1)N.CCOC CCCCCCC(F)C(=O)NCC(O)CCNC(c1cn(C)[nH]c1=N)=O N1(C(C2C(NC(=O)NCc3cccc(Cl)n3)C2)=O)CCOC2CC12 N1(C(C2CC(OC)C2)=O)CCC(O)(C(C)CNC(C2(CCF)CC2)=O)C1 c1(NCC2CC(=C)C2)cc(=NCc2cc(Br)cc(C)c2F)[nH]cn1 c1(C(N(CC(CC)NC(C(CCC#C)O)=O)C)=O)c(C)c(C)cc(C)c1C N1(C(c2c(C)ccc(F)c2)=O)CC(C)N(C(=O)C=CC2CCCN2C)CC1C C1(C2CCN(C(C3(c4ccccc4)CC3(F)F)=O)C2)(NC(CNC(N)=O)=O)CC1 c1(C(C)(C)C)ccc(CNC(=O)CN2CCCC3(CC3)C2)c(Br)c1 C(C(C)(C(C)C)NC(=O)CO)NC(C1(O)CC(C(=O)OC(C)(C)C)C1)=O C1(NC(c2cccc(OC)c2O)=O)CCCC12CN(C(c1ncc(C)cn1)=O)C2 Cc1ccc(C(=O)Nc2ccc(C(N3CCCNCC3C(N)=O)=O)nc2)c(O)c1 C1(S(C)(=O)=O)(C(=O)NC2CN(C(C(CC)C(=O)OC)=O)CC2C)CCCC1 c1(CN2CC3CN(C(=O)Nc4ccc(OC)cc4)CC32)ncc(OC)c(Cl)n1 C1(C(=O)NCCC(=C)C)COC(CNC(c2c[nH]c(C(N)=O)c2)=O)C1 C12(C(=O)NCCC3CN(C(C(C4CCC4)OC)=O)C3)C=CC(CC1)C2 c1(CC(=O)NC(C)(C(=O)Nc2cnc(F)nc2)C2CCC2)cccc(F)c1F CC(C)C(C(=O)NCCN(C(C1CC(F)C(=O)N1)=O)C(C)C)C1CCC1 Nc1cc(Br)cnc1C(=O)NC1CCCN(C(C2(CO)CC(F)(F)C2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1COCCN(C(C2CCOC(C)(C)C2)=O)C1 N12CCN(CC1)CC2=O.C1(C)(C(=O)NC(C)CS)CC2(CC2)C1.CCC(C)OC C(=O)(C(Cc1cnc[nH]1)NC1(COC)CC1)NC1C(COC)C1 c1(C(N2CCC(NC(c3c(C)noc3C)=O)C(O)C2)=O)cc(Cl)cc(Cl)c1O Cc1cc2nc[nH]c(=NCC3CC(CNC(c4ccoc4C(C)C)=O)CO3)c2[nH]1 Cc1ocnc1C(=O)NC(C1(O)CN(C(c2sccc2C(F)F)=O)C1)C CCC(F)(C(=O)OCC)C(=O)N1CC2CC1CC2NC(=O)CCC(C)C C=CC(C)(C)CC(=O)NCC1CN(C(C2(NC(C)C)CC2)=O)CC1C(F)(F)F N1(C(C=CCC)=O)CCCC(CNC(=O)C#CC(C)(C)C)(NC(=O)C(F)(F)F)C1 Cc1cc(NC(C2CCCCC(=O)N2)=O)ccc1NC(=O)CS(N)(=O)=O C1(C(=O)NCC2CCN(c3snc(CCC)n3)CC2C)CCC2CCCCN12 N1(C(c2c(OC)con2)=O)CCCC(C)(C)C1C c1(C(=O)NCC(C2CC2)NC(c2csc(O)n2)=O)cc(F)cc(F)c1 N1(C(c2cn(CC=C)nc2)=O)CC(CNC(=O)CC2(C#C)CCC2)C(O)C1 c1(C(N2CCC(CNC(C(n3ncc(C)c3)C)=O)C2)=O)cn(C)nc1OC(F)F c1(OC)cc(F)cc(C(N2CCC(CO)C(NC(=O)C(O)C(C)(C)C)C2)=O)c1N C(C(C)(C(N)=O)NC(C1(CNC(c2cncc(N)n2)=O)CCCCC1)=O)OC C(=O)(CC(C)CC(C)(C)C)N(C)CC1N(C(Cc2cn(CC)nc2)=O)CCCC1 C1(CC(=O)NC(C(=O)NC(C)C)C)CCCN(C(=O)CC2C=CCCC2)C1 C1(N(C(=O)CSCCC#N)CC)CCN(C(=O)CCSC2CCCC2)C1 Cc1ccc(CC(C)(C)OC(C2CCOC2c2ccc(F)nc2)=O)cc1 C1(C(=O)NCCN(C(CC2(COC)CC2)=O)CC(C)O)CC2(CCCC2)C1 C1(C(N(C(CC)C)C)=O)CCC(C)(C)N(C(=O)CN(C)C(=O)OCC)C1.C(C)C C1(C(N(CC(CC)NC(=O)C=C(C)C(F)F)C)=O)(COC)CCCCO1 C(=O)(C1=NOC(C)C1C)NC1C(NC(c2c(C)n(C(C)C)nn2)=O)COCC1 CC1CN(C(C2CCS2(=O)=O)=O)CCCN1C(c1cnn2c1CCC2)=O CS(=O)(=O)c1ccc(Cl)c(C(=O)NCCNC(=O)C=CC(F)(F)F)c1 c1(C(=O)NC2C(NC(Cc3cccc(OCC(C)C)c3)=O)C2)n[nH]c2c1COC2 C1(C(=O)NCCCOCCOCCC=O)CN(C)CC(F)(F)C1.CCCC(=O)NCC c1(CC)ccncc1-n1cc(C2CCCN2C(=O)C(F)(F)c2cccnc2)nn1 C12(NC(C#CC(C)C)=O)CCCC1N(C(=O)CSCc1cscn1)CC2 CC1CC(CC(N2CCC2CN=[N+]=[N-])=O)CN1C(=O)Cn1cccn1 c1(C(CC)NC(=O)CC2CCCC2O)ccc(Br)s1 c1(OC)cc(C(=O)NC2CN(C(c3cn(C)nc3SC)=O)CC2F)ccn1 C#Cc1cnc(C(=O)NC23CCN(C(c4cn(C)cc4C)=O)CCC2C3)c(C)c1 N1(C(Cc2c(C)noc2)=O)CC2(CC2)CC1CNC(=O)C(C)Cc1ccco1 C1(NC(c2c(C#C)cnn2C)=O)CC2CC(C1)N(C(=O)CSc1cnn(C)c1)C2 C1(C(N(CCN(C(=O)CCCc2ccncc2)C)C)=O)C(C)(C)C1(C)C N1(C(c2c(O)ccc(C)n2)=O)CCCC2(C1)C(NC(=O)CC(F)(F)Cl)CCN2C C(=O)(CC(C)C(F)(F)F)NCC(C1CCC1)NC(c1cccc(C(C)=O)c1)=O CC(CC(=O)NC1CCCC1CF)NC(C1(Cc2ccccc2)CCOC1)=O n1(CC)ncc(NC(C2(OCC(CCC)C3C(C(=O)NSC)C3)CC2)=O)c1C c1(CCC(=O)NCCN(C(c2c(NC)c(F)ccc2)=O)C)cccc([N+](=O)[O-])c1 c1(C(=O)OC)ccc(C=CC(=O)NC2(CCNC(=O)Cc3nccn3C)CC2)s1 n1(CC)cnc2c(NC(C)CC(N)=O)[nH]c(=NC(C)c3ccccc3)nc12 N1(C(c2nn(CC)c(O)c2)=O)CC(O)(C2(CNC(c3cnn(C)c3)=O)CC2)C1 C#Cc1cccc(CC(=O)NC(C)(CO)C(=O)NCC=CBr)c1 c1(C(=O)NCc2cn(CCN(C(=O)OC)CC)nn2)cc(Br)c([N+](=O)[O-])[nH]1 c1(C(=O)OC)ncc(NC(C2C=CCN2C(c2nccn2C)=O)=O)s1 c1(C(N2CC(CC(N3CCSCC3)=O)C2)=O)cc(O)cc(Cl)c1 c1(CN2CC(C(N3CC(CC)OCC3)=O)SCC2)nc(OC)cc(C)n1 C(=O)(CCCCCn1cc(CN2CCCCC2)nn1)N(C)CC1CCC1 Cc1nc(C(N2CCCC2CNC(c2ncc3ccccn23)=O)=O)c(=O)[nH]c1C c1(-c2nc(CCC(=O)NC(C)(CNC(=O)C=CBr)CO)on2)cccc(Cl)c1 CC(CCNC(=O)CCn1ncn(C)c1=O)CCNC(=O)C=C1CCC(C)C1 c1(C(CC2CC(F)(F)C2)N(CC)CC)cccc(NS(=O)(=O)C(F)(F)F)c1 C1(NC(c2cc(C)oc2)=O)C(C)CCN(C(=O)Cc2ccc(Cl)nc2)C1C N1(C(c2cc(C)c(O)nc2)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CC2(C)C1 c1(C(=O)NC(CNC(C(C(=O)OCC)OC)=O)CCOC)ncc(Cl)cc1Cl N12CCC3(CC3C1=O)C2.C1(C2N(C(CC3(COC)CC3)=O)CC2)CCCCC1 C1(NC(Cn2cccc(C(=O)OC)c2=O)=O)CCCN(C(=O)CC2CC2)CC1 c1(CCC)ccc(C(=O)NC(C2CCN(C(c3cc(C(N)=O)co3)=O)C2)(C)C)[nH]1 CC1(C)CC(CO)(CNC(=O)CC(CNC(=O)CCC2CCCO2)C2CCCO2)C1 N1(C(C(C)N(C(c2c(C(C)C)noc2)=O)C)=O)CC2(CCCC2)C1 N1(C(CNC(=O)COCC2CC2)C2CCC2)CCCCC1.C1CC(CBr)C1 C1(CC(=O)N(CCCC(=O)NCC2(OC)CC2)C)CC2(CCC2)C1 C=CCN(Cc1cccc(Br)c1)N1CCCC(C(=O)NC)C1 CN1CCN(C2CC2C(=O)NC2(CO)CN(C(C34CCC(CC3)C4)=O)C2)CC1 C(CCC(=O)NC(C1CC(n2cccn2)C1)=O)C1(NCC(C)(C)C)CCC1 c1(C(N2CCN(C(c3c(C)cc(C)o3)=O)CC2)=O)cccc2ncnc(O)c12 C(=O)(C(C)(C)C(=O)NCc1cc(Cl)sc1Cl)NC(C)CCN(C)C O=C1CC(C(=O)N2CCC2C(N2CCN(c3ccncc3)CC2)=O)=CC=N1.C(=O)N CCCC(F)C(=O)N1CCCC1CCNC(=O)CCC1CC(F)(F)C1 C(C1=CCN(C(c2ccn(CC(F)F)n2)=O)CC1)NC(C(C)(C)c1cc[nH]n1)=O C(C)(C)(CC(F)C(=O)N1CC(n2cnnc2)C1)NC(C(Br)=C(C)C)=O C(=O)(C1=C(C)CN(C(=O)C(=O)NCc2cn(C3CC3C(C)C)nn2)CC1)OC CCCCCC(C)CC(=O)NC(c1ccnn1C)C(=O)NCc1cn[nH]c1 C1(NC(CC2(C#N)CC2)=O)CC(C)(CNC(=O)CCC2CCCCO2)C1 C1(N(C(C(n2c(C)cc(C)n2)C)=O)C)CCN(C(=O)C#CC2CC2)CC1C C(=O)(C(C)(O)C(C)(C)C)N1CCC(CN(C(Cc2c(OC)ccnc2)=O)C)C1 c1(OC)ccc(CC(N2CCCC(C(C)SC)C2)=O)cc1S(N)(=O)=O c1(N2CCCC(NC(c3scc(C)c3)=O)C2C)ncnc2sc(C(C)(C)C)cc12 N1(CC(C)NC(C=C(C)C(C)C)=O)CCN(C(c2ncc(Br)cn2)=O)CC1 N1(C(CCC(=O)NC)=O)CCCC(C)(CNC(=O)CC2(OC)CC2)C1 C1(NC(CCC)=O)CCC(C)N(C(=O)Cc2cccc(C(F)(F)F)n2)C1 c1(C(=O)NC(CCCNC(C(CC(C)C)OC)=O)(C)C)cc2cn[nH]c2cn1 CCCC(C(O)C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CN=[N+]=[N-] CCCCCC(C(=O)NC)NC(C1CN(Cc2c(OC)cccc2F)C1)=O N1(C(c2cc(C)ncc2C)=O)CC2(CCCC2)C1C(=O)NCCC(C)N1CCC1 c1(-n2cc(CCOC)nn2)cccc(C(=O)NC2(C)CCSCC2)c1 c1(CCC)cc(C(N2CCC(O)(CNC(c3cc(SC)c(C)o3)=O)C2)=O)nn1C n1(CC)nnnc1C(c1nc(C)cs1)NC1(c2ccccn2)CCC1 C=CCCCC(=O)NC(c1cccc(Cl)c1)CNC(c1sc(=N)[nH]c1C)=O c1(NC(=O)OC(C)(C)C)cc(NC(=O)C(c2cccc(Br)n2)(F)F)cc(Cl)c1 C(=O)(CC1OCc2ccccc21)NC(C)CC(C)C.C1CCCC2CN(C2)C(=O)N1 N1(C(C2(C=C)CCN(C(c3n[nH]c(C)c3C)=O)C2)=O)CCCCCCC1CC c1(C(CCOC)NC(C2CC(CSC)C2)=O)cn2ccsc2n1.[nH]1cncn1 C#CC1(C(=O)Nc2ccc(OCF)cc2)CCN(C(=O)C2=NOC(C)C2)C1 C1(CC=C)(NC(C2CCC(C(N)=O)O2)=O)CCCN(C(c2cc(C#N)cs2)=O)C1 N1(C(C)C)CCCCN(C(=O)CC2CCCC(NC(=O)CN3CCCC3)C2)CC1 c1(C(N2C(CNC(=O)CC3(O)CC3)CCC2)=O)ccnn2ccnc12 n1(CC(C)CO)nc(CCN(C)C)nc1-c1cn(-c2ccccc2)nn1 C1(CO)CCN(C(C)=O)C12CCCC2.c1(CCC)ncc(C(=O)OC)s1 Cc1oc(C(C)C)cc1C(=O)NC1CC1CNC(=O)C(c1ccccc1Cl)O C1(C)(CNC(c2n(C(C)C)nnn2)c2cn(C3CC3)nn2)CCC(=O)NC1 c1(CNC(CNC(c2nc(C)no2)CC)=O)cc(-c2cccs2)[nH]n1 c1(OC)cc(CC(=O)NC2CN(C(=O)CCCCCF)C2)cc2c1OCC2.C(=O)OC C1(C)(CNC(C#CCNC(c2n(CC)ccc2)=O)=O)CCCCC1O C(C)(CCC#N)(c1nnnn1-c1cccc(Cl)c1)NC(c1scc(C)n1)C CN1CC(O)CCC1C(=O)NC(C)(C)COC1CCN(C(=O)CN(C)C)CC1 c1(C(N2CC(CC=C)(NC(c3ccn(C)c3C)=O)C2)=O)cnc(O)cc1C c1(CC)ccc(C(=O)N(C)CC2COCCN2C(c2cscc2SC)=O)cc1 CN1C(=O)C(=O)N(CC(=O)NCC2(C)CCCN2C(c2ccno2)=O)C1=O C1(CCNC(CCOCCCNC(C(C2CCCCC2)C)=O)=O)CCCOC1 Cc1nnc(CCC(=O)NC2(C)CC(NC(C3CNC(=O)N3)=O)C2)n1C c1(CNC(CCCOC)(C)c2nnnn2C)ccc(OCc2ccccc2)c(F)c1 N1(CCC)CCC(C(=O)NC(COCC)C(=O)NCCC2CCC3CC23)CC1 c1(-c2cc(C(=O)NCC3C(NC(=O)CC4CSCCS4)C3)on2)ccc(F)cc1 Cc1c(C(=O)NC2CN(C(C3CC3C)=O)C2)oc2ccccc12 Cc1nc(C(=O)NCC(C2CCCN2C(=O)CCCC#N)(C)C)c(C)o1 N1(C(CC)=O)CCN(C(c2ccc(SC(F)(F)F)o2)=O)CC(C)(F)C1 N1(C(c2c(OC)nsc2)=O)CCCC2CN(C(=O)CCc3cscn3)CCC12 c1(C(=O)NC2C3CN(C(COCCCOC)=O)C(C3)C2)nccc2occc12 C(=O)(C(CO)C(C)(C)C)N(CCC=C(C)C)NC(=O)CCCOC(C)(C)C c1(C(N2CC(N(C(C=CCC)=O)C)C(F)C2)=O)ccc2ncccn12 N1(C(c2cc(Cl)nn2C)C(=O)NC(C)C)CCC2(CCC(=O)NC2)C1 c1(NC(CCCN)C(=O)O)ccc2ccncc2c1[N+](=O)[O-] c1(C(=O)NC(CNC(C2(CCOC)CCC2)=O)CO)noc2ccccc12 c1(C(=O)NC(C)CCNC(C2CCCC2)=O)ncc(-c2ccncc2)s1 C(C(C(=O)NC1(CNC(C2CC2c2cccs2)=O)CC1)c1ccccc1)N(C)C C1(C(NCP(C)(C)=O)=O)CCCC(N(C)C)C1.C12(CC1)C(C)(C)NC2=O C1(NC(c2cc(C(N)=O)no2)=O)CCSC12CN(C(C1CCOCC1)=O)C2 c1(NC(c2ccc(Oc3ccc(C#N)cc3)nc2)=O)ccc2cnoc2c1 C1(CC)CCN(c2cc(N3CCOC(C4CC4)C3)nc(C)n2)CCO1 c1(CNC(C(=O)NCCNC(=O)CC2CCC(O)C2)=O)ccc(F)c(F)c1 CC(Cc1cnc[nH]1)C(=O)NCC(C)CNC(=O)COC1CC1 C1(NC(C(CC#C)C)=O)CCN(C(c2cc(OC)c(Br)cc2F)=O)CC1(C)C S1(=O)(=O)C=CCC(CC(O)(C)C(F)F)C(=O)N1 CCCC(=O)N(CC(=O)NC(c1ncc[nH]1)CO)CC(C)C O(NC(=O)C(CC)N(C)C(c1nc(CC)oc1C)=O)C(C=C)C Cn1nccc1C(F)=CC(=O)NC1CC1CNC(c1cc(C(N)=O)co1)=O C1(N=c2[nH]nc(SC)s2)(CCOC)CCN(C(C23CCCC(C2)OC3)=O)C1 C(CCCc1ccccc1)(C(=O)NCC(=C)C)N(C)CC1CC(=C)C1 C(C(N=c1ccc2nnc(-c3cc(C)cc(C)c3)n2[nH]1)C(F)(F)F)OCC C1(NC(C(c2n(C)ncc2)O)=O)CCCN(C(C2CC=CC2)=O)CC1 N1(CCNC(COCC(=C)C)=O)CCC(NC(=O)C(C)C2CCCO2)CC1 c1(C(=O)NC(C(C)NC(=O)CCC2CCCCC2)(C)C)cnc(O)c2cncn12 c1(C(=O)NCC(=O)NCC(C)CNC(C2CCOC2)=O)cccc(Cl)c1 C1(C(=O)NC2(C)CCN(C(c3cc(C)nn3C)=O)CC2)CC12CCC(C)(C)CC2 c1(C(N(C2CN(C(=O)CCc3nccn3C)C2)C)=O)cc(C(F)(F)F)cnc1N c1(C(=O)NC(CN(C(c2c(CC)onc2)=O)C)CC)ccc(C(C)CC)nc1O Cc1ccc(C(=O)NC(C2CCCN2C(c2cc(C)sn2)=O)C)c(O)n1 c1(C(N2CC(C)(NC(C3CC34CCCOC4)=O)C2)=O)csc2c1CCCC2 c1(C(=O)OC)cc(F)c(S(=O)(=O)NC(C)C(c2cc(F)cc(F)c2)O)c(Br)c1 C(=O)(CCS(=O)(=O)C(F)(F)F)N(C1CCCCN(C(C(CC)(C)C#N)=O)C1)C C1(NC(c2cccc(Cl)c2Cl)=O)CN(C(c2cc[nH]c2)=O)CCC12CCOCC2 c1(C(=O)NCCNC(Cn2ncc(C(=O)OCC)c2)=O)ccc2oc(C)nc2c1 C12(O)CCCN(C1)C2=O.C1(CC)(CNC(=O)CC(Cl)Cl)CCCCC1 c1(C(=O)NC(CNC(C2(CC)CCCC2)=O)(C)CO)ncnc(C)c1C N1(C(c2ccc(C)s2)=O)CC(C)OC2(CCN(C(C3CSC3)=O)C2)C1 N#Cc1ccc(=NCC(=O)NCC2CC2NC(c2ccccc2C(F)F)=O)[nH]c1 N12CC3(CC3)CC1COCCC2.C(=O)(CCC(F)F)NCc1nc(CCCC)on1 n1(CC)cnc2c(N(C3CCCCCC3)C)nc(NCC(CCC)CCO)nc12 C12(NC(CCCCSC)=O)CC(CNC(=O)CSC(F)F)(C1)OC21CCC1 c1(C(C)(C)C)cc(C(=O)NCC(F)(F)Cn2cc(CC3CCOC3)nn2)cs1 CCCCC(CC)CCC(=O)N1CC(COC)(NS(=O)(=O)c2ccccc2Cl)C1 c1(C(N2CC(CCNC(C=CSC)=O)OC(C)C2)=O)cc2cc(C)ccc2o1 CC1=C(C)CC(C(=O)N(C(CNC(=O)CS(N)(=O)=O)C2CC2)C)CC1 N1(C(CCc2c[nH]c(C)cc2=O)=O)CCN(C(=O)CCCS(C)(=O)=O)CC(O)C1 N1(C(CN2CCN(C(C(c3cccnc3)C)=O)CC2)=O)CCC2(CC1)CC2 c1(CC)ccc(NC(c2nnnn2C2CC(CC)C2)c2nncs2)c(CC#N)c1 C(=O)(C=CS(C)=O)NCCC1CCN(C(C2(CCOC)CCC2)=O)C1 C1(C(=O)NCC2CC2C2CCCO2)CN(C(=O)CC2(O)CCC2)CCO1 CC1=C(C(=O)NC(c2cccc(C(=O)O)c2)CC(=O)O)Cn2ncnc2N1C c1(C(N2CCC(C(F)F)(CNC(C3CC=CC3)=O)C2)=O)nccc2ncccc12 N1(C(C2(c3ccc(-c4ccc(B(O)O)cc4)cc3)CC2)=O)CCCC2(CCOC2)C1 c1(C(=O)NCC(C)N(C(c2ccc(F)c(O)c2)=O)CC)cc2c(nn1)CCCO2 CC1(C)CC(=O)NC1CNC(=O)C(C(C)(C)C)NC(c1ccc(F)cc1F)=O C(=O)(C(C(C)C)NC(C)=O)NCC=CCC(=O)NCC(CC1CC1)OC N1(C(c2nc(OCC)oc2)=O)C2CCC1C1CC1(NC(=O)C(F)n1ccnc1)C2 C1(CNC(C2CN3CCCC2C3)=O)CN(C(=O)C2CC2)CCC1(F)F N1(C(CC(CC)N(C(=O)C=CCOC)C)=O)CCCC2(CC1)CC2 N1(C(C(C)NS(C)(=O)=O)=O)CC2=C(C1)CN(C(c1c[nH]ccc1=O)=O)C2 N1(C(C(CC(C)C)=O)=O)CC2(CCCC2)C1CN.C12CCCCN1C(=O)C(C)S2 c1(N2CC(CNC(=O)OC(C)(C)C)C3(C2)CC3)nc2ccccc2s1 C1(c2ccccc2)(C(N(CC(C)(C)C)CC(C)C)=O)CC2(CC2)C1 C1(OC)CC(CNC(=O)CCCc2cccs2)N(C(c2n[nH]c(C)c2O)=O)C1 CC1C(NC(=O)CC2(C)CCC2)CCCN1C(c1csc(C(C)O)n1)=O C1(C)(CNC(c2c(OC)csc2)=O)CCN(C(C2(C)CC(O)C2)=O)C1 c1(OC)cc(C(N2CCCC(NC(=O)C(=O)O)C2)=O)cc([N+](=O)[O-])c1 C1(C)(C(=O)NC(C2CCN(C(C34CC3CNC4=O)=O)CC2)C)COC(=O)C1 C1(N(C(C)C(=O)N2CCCC2)C(COCCOC)=O)CC(C)CC(C)(C)C1 C(=O)(CCCCCO)N1CCC(N(CC#C)C(C2CC2(Cl)Cl)=O)CC1 C1(C(=O)NCc2cn(CCO)nn2)CCN(C(=O)C=Cc2cscn2)C12CCC2 Cc1cccc(COCC(=O)NC(C2CCN(C(C3CCCC(=O)O3)=O)C2)C)c1 Cc1ccnn1C(C)C(=O)N(C1CCN(C(=O)CCc2cnn(C)c2)C1)CCO N1(C(c2nnn(CC)c2C)=O)CC2CC1CN2C(=O)C(c1c(Cl)cccc1Cl)C CCC(C)(CCNC(c1cnc(C2CC2)o1)=O)NC(c1cc(Cl)ns1)=O C1(C(=O)NC2C=CC(C(=O)NC)C2)CCN(C(=O)c2cc(C)cc(O)n2)O1 CCCC(C)(C)CC(=O)N1CCN(C(c2cc(C#N)ccc2C)=O)C(C2CC2)C1 C1(NC(CCOCC#C)=O)CCC2(CC1)CC2NC(=O)C(C(C)(C)C)SC C(C)(C(=O)N1CC(CNC(C2CC(O)C2)=O)C1)N(CCC)C(=O)OC(C)(C)C N#Cc1cccc(CCC(=O)NCCC2CN(C(C3CCSC3)=O)CCCO2)c1 c1(C(N2CCCCC2C(C)CO)C(=O)NCCOC)cc(C)ccn1 c1(C(=O)NCCOC2CCN(C(C(CC)C(C)C)=O)C2)ccc2nnnn2c1 n1(CC(C)C(=O)NCCNC(=O)CCC2(O)CCOCC2)ccc2ccccc12 CC1=NOC(=O)C1CC(N1CCN(C2CN(C(c3c(F)cnn3C)=O)C2)CC1)=O C1(C(C)C)CN(C(c2[nH]cnc2C)=O)CCN1C(C1CC1(C)Br)=O CCC(O)C(C)C(=O)NCC(F)(F)Cn1cc(C2(O)COC2)nn1 N1(C(C2(C)CC2)=O)CCCC(C2(NC(C3CN(CC(F)(F)F)C3)=O)CC2)C1 N1(C(C(CCC)OC)=O)CC(NC(=O)CCc2ccc(Cl)s2)CC(F)C1 c1(OC)c(F)ccc(F)c1CN1CC(NC(C2CCCS2)=O)C(F)(F)C1 C(=O)(C1CCCc2ncnn21)Nc1ccnc(F)c1.CC1CCC2CN1C2 c1(C(N2CCCC(C(=O)NC(CSC)CO)(CC)C2)=O)cc(C)cc(C#N)c1 C(CCC(C)C(=O)NCC(C1CCN(C(=O)C=C2CCN(C)CC2)CC1)C)OC c1(OC(C)C(N2C3CCC2C(NC(=O)C(F)(F)CO)C3)=O)ccc2c(c1)CCC2 N1(C(C(=O)Nc2cc(C(=O)OCC)sc2C)=O)SC(=N)NC(C)(C)C1 C1(C(=O)NC(CC(=O)N(C2CCCCC2)C)C2CC2)CC2(CC2)CO1 C1(F)(CNC(c2n(C)nc(O)c2)=O)CCN(C(C2CCOC(C(F)F)C2)=O)CC1 CC1(C(N2CCOC(CC(=O)NC(CO)C3(C)CC3)C2)=O)CC(C#N)C1 N1(C(C2CC(CCC)OCC2)=O)CC(C2(NC(=O)CC(=O)NC)CC2)C1 c1(CNC2(c3n(CC)nnn3)CCC(C)C2)cccc(C(F)F)c1F N1(C(C2NC(=O)CC(=O)C2)=O)CC(C(=O)Nc2cnn(C3CC3)c2)CC12CCC2 Cc1ccc(C(=O)NC(CO)C(C)NC(=O)CC2COCC2O)cc1N N1(CC(=O)N(CC)Cc2cnn(C3CCOCC3)n2)CCN(C)C2(CCOC2)C1 C1(C(=O)NC(CC#C)C)(CC)CCCN(C(=O)C(CN(C)C)N(C)C)C1 N1(C(COCCCC#C)=O)CCCC(O)(CNC(C2CCCC(=O)N2C)=O)CC1 CC1(C)C=CC(OC2CC(OCC(=O)NC3CCCC3)C2)CC1 C(=O)(CC(C(C)C)NC(C1CC(C)=NO1)=O)N(CCCC)C Cc1[nH]nc2cc(C(=O)NC3CC3NC(c3c4c(nn3C)CCSC4)=O)ccc12 C1(NC(C(C2CCC2)OC)=O)CN(C(=O)C(C)(C)CF)CC1c1ccccc1F C1(NC(COCc2cc(C)on2)=O)CC12CCN(C(=O)CCc1cccs1)C2 CCC(C)(CCC(C)C)C(=O)NC(C)CCN(C)C(c1ccccc1CC#N)=O c1(C(N2CCC(C)(CNC(CCCOCC)=O)C2)=O)cc(C)ccc1N c1(NC(=O)NCC(C)CNC(=O)CNc2ccccc2)ccn2ccsc12 O=C1CC(NC(=O)CN(C(=O)CCn2cccn2)C2CCC2)CN1 c1(C(=O)NCC(C)CNC(C2CC3C=CC2C3)=O)ccc(C(F)C(F)(F)F)cc1 C1(C(=O)NC2C(N(C)C(c3cc(C4CC4)sn3)=O)CCOC2)COCCC1(F)F C1(NC(c2c(C)ncnc2C)=O)CCC2CCN(C(=O)C(C)n3ccnc3)C12 C1(C(=O)NCC(CC=C)(C)C)CC(F)CCN1c1c(NC)cccc1 C1(NC(COC(CC)C)=O)CN(C(=O)C=Cc2ccc(Br)o2)C(C)(C)C1 C(=O)(CCCCC(F)F)NC12C(CN(C(C(c3ccc(OC)cc3)(C)C)=O)C1)C2 C12CN(CC1C(C)C)C2=O.c1(C(=O)N)cc(CO)[nH]n1.C(C(=O)OC)(C1CC1)SC c1(C2C(C(=O)NCC(CN(C(=O)Cn3[nH]cnc3=N)C)O)C2)cnn(C)c1 C(N(C)N1CC(C)(OCCOCCOC(C)(C)C)C1)c1cccc(C(=O)OC)n1 C1(C(=O)NC(CN(C(COCCOC)=O)C)C)(COC)CCCO1 N1(CCC)CCCC(C(=O)N(C(C)CCNC(=O)CCc2cc(Cl)cs2)C)C1 C1(CNC(CS(CC)=O)=O)(OC)CCN(C(c2c(OC)ccnc2F)=O)CC1 C1(NC(c2nc(CNC(CN(C(=O)OC)C)=O)oc2)=O)CC(=O)N(O)C1 C1(CNC(C(C(=O)OC)(C)F)=O)CC2CCC(C1)N2C(C1(CC2CC2)CC1)=O Cc1ccc(C)n1-c1ccc(C(=O)NC2(CN(C)C(C3CC34CC4)=O)CC2)cc1 N1(C(=O)Cc2cn[nH]c2)CCC(C2CCO2)CC1 CCCC(C(=O)NC(C)(C)CCNC(=O)CC1CCC(F)(F)C1)OCC C1(NC(c2ccc3nccn3c2)=O)CS(=O)(=O)C2CN(C(c3cc[nH]c3)=O)CC12 c1(C(N2CC(NC(c3cc(-c4ccncc4)no3)=O)C2)=O)cc(Cl)cc(Cl)c1Cl N1(C(=O)NCc2cc(CC3CCCO3)ncn2)CCN(c2ccccc2)C(=O)C1 c1(C(N2CC(N(C(c3c(C)noc3)=O)C)C(F)C2)=O)cccc(C(F)(F)F)c1Cl Nc1c(NC(=O)NCCC#CBr)cc(F)cc1[N+](=O)[O-] c1(C(=O)NCC2CC(NC(c3cc(C)sc3C)=O)CC2O)ccsc1S(C)(=O)=O N1(C(C2N(C(=O)COc3ccsc3)CCC2O)=O)CCOCC(C2CC2)C1 C1(C(=O)NC(CC)CCCO)C(C)OCCN1C(C1CCCC1O)=O C1(n2c(CC(C=C)CC)nc(COC)n2)CCC(C)(C)CC1 c1(NCC2CC(CC)OCC2)cccc(OC)c1Cl CC1CN(C(c2cc(O)cc([N+](=O)[O-])c2)=O)CC2(CCN(C(=O)C(F)(F)Br)C2)O1 c1(C(=O)NC(CCN(C(C2CC(SC)C2)=O)C)(C)C)cnc(C)nc1 C12(CNC(C3CC3F)=O)CCC(C1)N(C(=O)Cc1csc(N3CCNC3=O)n1)C2 c1(C(=O)NC(C2(N(c3ccccc3)C(=O)CC3CC3)CC2)C)cncc(C(F)F)c1 N1(C(C=Cc2occ(C)n2)=O)CCC2C(NC(c3ncccc3Br)=O)CC12 CC12CC3CC(CC(C(N4CCOC(CNC(=O)C5=NOCC5)C4)=O)(C3)C1)C2 c1(C(=O)NCC(CO)NC(c2ncc(C#N)cc2Cl)=O)cnc2[nH]c(O)nc2c1 Cc1csc(C(=O)NCC2CCCC2NC(c2cc(CCO)on2)=O)c1C CC1(C(=O)OC(=O)C(=O)OCCOc2ccccc2)CC2C=CC1C2 c1(NCC2CN(C(Cc3cc(C)cc(C)c3)=O)C2)ncc([N+](=O)[O-])cc1Cl Cc1c(-c2nnc(N3CCOC(C4CCOC4)C3)n2CCC#N)ccn1CCO C1(c2n(CCC)nnn2)(NCc2nnc(CO)s2)CCS(=O)(=O)CC1 CCC(CC)C(C)C(=O)NCCC1CCN(C(c2nocc2C(C)C)=O)C1 N1(C(C(C)=C(CC)C)=O)CCCOC(CNC(=O)CCC2CC2(C)C)C1 N1(C(C(C)c2ccco2)=O)CCCN(C(c2ncoc2C2CCC2)=O)CCC1 C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2sc(CC)nc2C)=O)CC1O Cc1snnc1C(=O)NC1CCC(CCNC(=O)Cc2ccc(Br)s2)C1 c1(C(N(C2C(C)CCN(C(CCC=CC)=O)C2)C)=O)cccc2c(C)ccnc12 Cc1ccc(F)c2[nH]c(C(=O)NC3CN(C(=O)CCC4(C)CC4)CC3C)cc12 C=CC1(C(=O)NCC2(C)CCC(=O)N2)CCN(C(c2c[nH]nc2Cl)=O)C1 CN1CCN(C(C23CC(c4ccccc4)C2C3)=O)CC1c1cccs1 Nc1cccc(C(N2CCCC(CNC(c3cc(=O)cc(Cl)[nH]3)=O)C2)=O)c1N c1(CC)noc(CC)c1CC(=O)N(C(CNC(C1(C)CC(F)C1)=O)C1CC1)C N1(C(CCCC(C)C)=O)C2CCC1CC(NC(c1coc(Br)c1)=O)C2 C(=O)(C(CC(C)C)CC(C)C)NC1C(CNC(C(C=C)(C)C)=O)CCC1 C12(C(=O)NC3CC(N(C(c4c(C)nc(C5CC5)[nH]4)=O)C)C3)CCCN1CCC2 CC1COCC(CC(=O)NCc2cc(C(=O)N(C)CCN3CCCC3=O)on2)O1 C1(CN(c2nnc(-c3cccc(O)n3)n2CCC#N)C)CCc2c[nH]nc2C1 c1(OCC(=O)NCC2(NC(C(CC)C)=O)CC2)cccc(Cl)c1.C(=O)(CO)CCOC C12(CC)COC(C(=O)NC3CC(CNC(C4C(C=C(C)C)C4(C)C)=O)C3)(C1)C2 N1(C(C=CCCC)=O)CC(NC(C2(CC)CCOC2)=O)CC(C)C1 N1(C(CN(C2CC2)CC)=O)CC(NC(=O)CN2CCCC2CO)C2(CCC2)C1 c1(C(N(C(CNC(c2ccc(OC)cn2)=O)C)C)=O)ccc2ocnc2n1 c1(C(C)NCC(c2c(C)nns2)OC)ccc(Oc2cccc(F)c2)nc1 C(=O)(C1=NOC(C)(C)C1)NC(C)C(=O)NC(C)Cc1ccnn1C N1(C(CC2CC(CC)OCC2)=O)CCCC2(NC(=O)C(C3CC3)C3CC3)CC2C1 C1(C(N2CC(C(C(C)C)O)C2)=O)CCN(C(C2CC3CCC3C2)=O)CC1C c1(NC(C2CCCN(Cc3c(Cl)ccnc3Cl)CC2)=O)cc(CO)cc(F)c1 c1(NC(C2CC(CNC(C(C)n3ccnc3)=O)C2)=O)cncc(F)c1 c1(C(=O)NCC(=CC(N2C(C(=O)OC)CSC2)=O)C)ccc(C)c(C#N)c1 N1(C(CCSCCNC(c2c(CC)nn[nH]2)=O)=O)CCC(C)C(CO)C1 N1(C(CCNC(COC)=O)=O)CC2(COC(CNC(=O)Cc3cnsc3)C2)C1 Cc1ccc(C(=O)NC(C2CN(C(=O)Cn3cnc(Br)c3)C2)C)s1 C1(NC(CCOCCCCC)=O)(CC)CCCN(C(C2(CC3CCC3)CC2)=O)C1 n1(CC(C)C)[nH]c(CC(=O)NC2CN(C(=O)C(F)C3CCC3)C2)cc1=O C1(NC(c2ncccc2O)=O)CN(C(c2cnn(C3CC3(F)F)c2)=O)CC12CC2 CC1(NC(C2CCC(=O)N2)=O)CCN(Cc2nc(C(F)F)no2)CC1 CC1(C)C(C(=O)NC(c2ccc(OC(F)(F)F)cc2)CO)CC12CCN2 C1(NC(C(CC)C(C)C)=O)CC2(CCN(C(=O)C#CC3CCCO3)CC2)C1 c1(C(C)NC(N(Cc2ccc(OC)cc2)Cc2cccs2)=O)ccc(C#N)cc1 c1(C(N2C3C(CNC(C(CC)(C)O)=O)CC(CC3)C2)=O)ccc2cncn2c1C C=CC(C)(CC)C(=O)NCc1cccc(CNC(=O)Cc2ccno2)c1 N1(C(c2[nH]cc(C)c2)=O)CCN(Cc2cnn(-c3cccc(C#N)c3)c2)C2CC12 N1(CC#C)CCCC1C(N1CC(CNC(C2COCC2C(N)=O)=O)(OC)C1)=O C(=O)(C1=CCCOCC1)NCC(C)(CNC(c1cnc([N+](=O)[O-])n1C)=O)OC CC1C(C)N(C(C2CCC3(CC2)CC3)=O)CCN1C(c1cc(C(F)(F)F)n[nH]1)=O c1(C(N2CC3C(NC(c4cn(C)nn4)=O)C(C3)C2)=O)cccc2nnn(C)c12 c1(C(=O)NC(C)(C)CN2CCN(C(=O)C(F)C3CC3)CC2)cnc2[nH]cncc1-2 c1(OC)c(CC(N2CCC(C(C)NC(=O)CCOC3CC3)C2)=O)cccc1F CCCCS(=O)(=O)N1CCCC(C(=O)NC2(C)CCC2)C1 c1(C(N2CCN(C(C(CCC)C)=O)C(COC)C2)=O)sc(=NCC)[nH]c1C C1(NC(C2C(=C)CC2)=O)COCCC1C(=O)N(C)CCN(C)CCO c1(C(=O)NCC(CNC(=O)CCc2cncs2)O)ccc2nsnc2c1 C(C(=O)NN1CCCC1C(=O)NC(C)CN1CCCC1=O)SC(C)C C(=O)(CCCCCCCCC1CC1)NC1C(NC(C(C)(C)OCC)=O)CCC1 c1(NC(CC)Cc2nnnn2C2CCCC2)ccc(OC(F)F)cc1.c1nnn(C)c1C N1(C(C2(C)CC(=C)C2)=O)CCC(NC(=O)CC2(C#N)CCC2)C(C)C1 C#CC1(NC(C2CC3(CC(NC(c4ccnnc4)=O)C3)C2)=O)CCCOC1 c1(OC(C)C)cccc(CCC(=O)N(CC(C)CNC(=O)C(C)CN(C)C)C)c1 C1(OCCOC)CN(N2CC(CO)CC2C)CC2(CCC2)C1 O=C1CCCCC(C(N2CCCN(C(C3CCC(F)(F)C3)=O)CC2)=O)N1 C1(COC2CCN(C(CCOC)=O)C2)CCC2(CC1)CC2 CC1(C)CC(C(N)=O)CCN1C(=O)CC(O)CNC(c1cccnc1)=O CS(=O)C=CC(=O)N1CC(NC(=O)Cc2cccc(C(F)(F)F)c2)C(F)C1 c1(CSCCN(CCOC)C(=O)NC2CC3CCC2C3)cccc(Cl)c1 C(=O)(CC1CCOc2ccccc21)N1CC(O)CC(NC(COCCC=C)=O)C1 C(=O)(CC(O)CC)N(C1CCN(C(C2CC2F)=O)CC1)CCC N12CCC(CC1C)NC2=O.C(=O)(C=CC=CC)N.C(C)(Cl)=C c1(NCc2nnc(CC)n2C)[nH]c(=NC2CC3(CC3)C2)nc2sccc12 N1(C(c2cncnc2)C)CCC2(CC1)CN(c1ncnc(C(C)(C)C)n1)CCO2 CCCC(C#N)C(=O)NC(CC1CCCC1)C(=O)NC(CN(C)C)CC N1(C(c2n(CC)nc(C)c2)=O)CC2CCC2(NC(c2ccoc2Cl)=O)C1 C(=O)(C(CC(C)C)N1CCCCC1=O)NC1C(NC(C2(SCC)CC2)=O)COC1 c1(C(N2CCC(NC(c3cc(Cl)c(F)c(Cl)c3)=O)CC2)=O)cc(F)cc(F)c1F c1(C(=O)NCC2(F)CCN(C(C(CN(CC)CC)F)=O)C2)ccc2nn[nH]c2c1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1C C(=O)(CC(C)(C)C)NC(C1CCN(Cc2nccs2)CC1)C(C)C CC(C)C(CNC(=O)C(C1CCOCC1)F)C(=O)N(C)CC1CCCS1 c1(C(C(=O)NC(C2CCCN2C(C2CC(C)(C)O2)=O)C)(F)F)ccc(Cl)c(Cl)c1 C1(C(C2CCOC2)SCC(=O)NCC2CCCO2)CCN(Cc2cccnc2)CC1 C(=O)(C(CCCC=C)NC(=O)C(C)OC)NC(CC#C)C(=O)OCC c1(C(=O)NCC2N(c3ccnc(SC)n3)CCCC2)c(F)cc(Cl)cc1Cl C1(CC)CN(C(c2ccc(CF)cc2)=O)CC1NC(c1cc(C#N)c[nH]1)=O N1(C(CC2CCCC(C)O2)=O)CC2(CC(NC(=O)C=Cc3cccnc3)C2)C1 C1(C(=O)NC(COCC)C(C)C)CCCCN(C(=O)C(C)(C)O)C1 C=CCC(CC(=O)NC1CCOCCC1)NC(c1ocnc1C)=O c1(CC(=O)NC2C(CNC(C(COC)C)=O)CCC2)ccc2c(c1)CCN2C c1(-c2cccc(C#N)c2)n[nH]c2c1CN(Cc1ncco1)CC2 C(=O)(C1=CC2CCC=CCCC12)NCCC1CN(C(c2c(C)cc(Cl)cc2)=O)C1 N1(C(CCOCCC)=O)CC2C(CNC(=O)CSC3CC3)C2C1 C1(NC(C(C)(C)CF)=O)CS(=O)(=O)CC1NC(c1nsnc1O)=O CCN=c1cc(-c2nc(C(O)Cc3cccs3)n(C3(C(N)=O)CC3)n2)cc[nH]1 CC(C)C(C(=O)NCC(C(=O)NC1CCC2(CCC2)C1)C(C)C)C(C)C C1(CNC(C(CCC)C)=O)CCCC2(CN(C(=O)CC3(COC)CCCC3)C2)O1 C=CCCC(C(=O)N1CCOCC1CN(C)C)NC(=O)C(F)CN(C)C C(=O)(NNC(=O)COCCCN=[N+]=[N-])NCC1C(C)C1 CC1CC(N=c2c([N+](=O)[O-])c[nH]c3ccc(F)cc23)CCN1C(C1CCC1)=O c1(-c2nc(CC(=O)NCc3c(C(C)O)cccc3)c(C)s2)cc(F)ccc1C C1(C(N2CCCC(N(CC#C)C(c3nn(C)cc3SC)=O)C2)=O)CC2CC(=O)C1O2 Cc1cc(C(=O)NCCOCC(=O)NCc2cc(C#N)c[nH]2)n(C)n1 N1(C(C(COCC)C)=O)CC2CCC2(C(=O)NCC2(CCOC)CC2)C1 C(=O)(CCCC(C)O)N1CCC(N(c2ccnc(C(C)C)n2)C)C1 N1(C(C(CC=CC)C)=O)CCC(NC(=O)C2=CCCO2)C1(C)C C1(CNC(C(CC)O)=O)CC(C)N(C(=O)Cc2ccc(Br)cc2)C1 CC(F)(C(=O)NCCC1CN(C(=O)CCCc2ccccn2)C1)C(F)(F)F c1(C(=O)NCCCCNC(=O)C(C2CCCCC2)F)n[nH]c2c1CC1CC21 C1(C(N(C2CN(C(CCCc3onc(CC)n3)=O)C2)C)=O)CCS(=O)(=O)C(C)C1 C(=O)(C(CC=C)C(C)C)N(CC(CNC(COCCCC#C)=O)(C)C)C C1(NC(C(COC)O)=O)CCCC12CN(C(=O)CCCCC(F)F)C2 Cc1csc(C(=O)NC2CCC2NC(C23C=CC(CC2)C3)=O)c1Cl CC1CN(C(C2CCCC(F)(F)C2)=O)CCN1C(=O)CN1C(=O)CN(C)C1=O CC1(C)OC(=O)C(CC(=O)NC2CC(NC(=O)CSc3nc[nH]n3)C2)O1 C12(OC)CCCCC(C(=O)NCCN(C(=O)C3=CCCOC3)C)(C1)C2 c1(C(=O)NC(C)CNC(c2ccc(C(F)(F)F)o2)=O)cc(Br)cnc1O c1(C(C)OC)nc(C)c(C(=O)NCC=CCNC(C2CCSCC2)=O)s1 c1(C(=O)NC(CC)CNC(c2cccnn2)=O)ccc2nc[nH]c2c1F N1(C(C(C)(C)OCCC)=O)CC2CC2(CN(C2COC2)C(=O)CC)C1 N1(CC(CN(CC#C)C(=O)OC(C)(C)C)O)CCN(c2ccccc2)CC1 N1(C(C)C)CCCC(C(=O)NC2CCN(CCc3nc(C(C)C)no3)CC2)C1 C(=O)(C1=COCCO1)N1CCC(C(C)(C)NC(=O)C(F)(F)c2ccsc2Cl)C1 c1(CC(=O)NC2CC2)cccc(-n2ncc(C3OCCO3)c2Br)c1 N1(C(c2csc(Cl)n2)=O)CCOC(C2CN(C(=O)C=CC(F)(F)F)C2)C1 C1(C(=O)NCC2=CCN(C(C3C(C)(CC)C3)=O)CC2)CC(c2cccnc2)=NO1 C=CCCCCC(=O)N1CCCC(N(C)C(C2CCCC2F)=O)CC1 C1(NC(c2ccc(C3CC3)o2)=O)CN(C(C2CC3CCC2O3)=O)CC2(CC2)C1 C(=O)(CC(C)C(F)F)NCC(CNC(CCc1c(OCC)cccc1)=O)CO C(C(Cc1ccccc1)C(=O)N1CCC(c2cncc(F)c2)C1)CO C(=O)(N=c1cc(C)n(C)[nH]1)C1(CCNC(COC(CC)(C)C)=O)CCCC1 Cc1cccc(CC(N2CCC(NC(=O)CC3CCCCC3F)CC2)=O)c1F C12(C(N3CC(CCNC(C(C)n4ccnc4)=O)C3)=O)CCC(C(F)(F)F)(CC1)C2 C1(O)(CC#C)CCN(C(C2C3CC2N(C(C2CCC(F)C2)=O)C3)=O)CC1 C1(C#N)(C(=O)NCCN(CC(C)O)C(c2cn(CCC)nc2)=O)CCOCC1 C(CN=[N+]=[N-])(C(=O)NC(C)C(=O)N(C)C)NC(CSCCOC)=O C(=O)(C(CSC)C(C)C)N(CCNC(c1cn(CC(CC)O)nn1)=O)CC1CC1 CC(CN=c1[nH]c(N2CC3OC3C2)nc2c1COC2)c1ccncc1Br.CO C12(NC(c3ccc(F)cn3)=O)CCCCC1CN(C(C1CC3CCC1C3)=O)C2 c1(C(=O)OCC)sc(C(=O)NCCC(O)CNC(C2CC2F)=O)c2c1CCCC2 C1(N(C(Cc2scc(C)n2)=O)C)CN(C(=O)CC2CC3(CC3)C2)CC1(C)C c1(C(=O)NCCCNC(C2(F)C(C)C2)=O)cccnc1OC(F)(F)F.C1(O)CCCC1 n1(CC)ncc(C(=O)NCC2C3CN(C(=O)Cc4conc4C)CC23)c1N c1(OC)c(F)cc(F)c(CN2CCS(=O)(=O)C(CCNC(=O)CO)C2)c1[N+](=O)[O-] C(N=c1cc(-n2cccn2)nc[nH]1)C1N(CC2S(=O)(=O)CCC2)CCC1 C1(NC(CCCOCCOC)=O)CN(C(c2n[nH]cc2Cl)=O)CC1n1cccn1 C12(CCNC(CC3(OC)CCC3)=O)CCC1CN(C(c1cc(Br)co1)=O)C2 c1(C(=O)NC(CC=C)CNC(c2ccncc2OC)=O)ccnc(OC)c1F C1(CNC(C2(CCC)CCC2)=O)CCN(C(=O)CCC=CBr)CC1C CS(=O)(=O)C1(C(N2CCCOC(CNC(c3cc(C#N)oc3C)=O)C2)=O)CCC1 c1(C(=O)NC(CNC(C(c2nc(C)sc2)=O)=O)(C)C2CC2)cc(C)cn1C c1(C(N2CCC(C)(C#N)C2)=O)ccn2ncccc12.c12cccc(c1)NC2=O N1(C(C(n2ccc(C(F)(F)F)n2)C)=O)CCC(N(CCO)C(C2CCC2)=O)CC1 C=CC(CC)CC(=O)N(C)CCNC(C1(c2c(F)cccc2Cl)CCC1)=O C(=O)(CCCN=[N+]=[N-])N1CC(C(N(CC(C)C(F)(F)F)C)=O)(N(C)C)C1 N1(C(C2CCC(=O)N2)=O)CCC(n2cc(COc3ccc(F)cc3)nn2)C(O)C1 c1(C(=O)NCC(CNC(C(COC)(C)O)=O)C(F)(F)F)ccc(S(C)(=O)=O)cc1 CCCCC(CC)CC(=O)NC(C)(C)CNC(=O)C=CC1CCC1.C(=O)(C=CCF)OC c1(C(N2CC3CC3(C(=O)Nc3cccc(Br)c3F)C2)=O)ccn2cncc2c1 N1(C(c2cnc(C(F)(F)F)s2)C(=O)NC(CC)(C)C)CC(C)SC(C)C1 N1(C(C2(C)CC=C(C)CC2)=O)CC2(CCC(CNC(=O)CN(S(C)(=O)=O)C)O2)C1 c1(C(=O)NC2C(CNC(c3occ(C(=O)OC)c3)=O)CC2)cccc(F)c1 Cc1cccc(Cl)c1CC(=O)NCCC1CN(C(C2CCN(C)C2=O)=O)CCO1 C=C=CCC(=O)NC(C)CCNC(C1CCC(C(F)(F)F)C1)=O C#CC1(C(=O)NCCN(C(=O)CC2CCCN2C(C2CCCCC2)=O)C)CCC1 O=C(CCCCCl)NCC1CC1(F)F C=CCCCCC(=O)NC1(CCNC(=O)Cc2sc(C)cc2C)CC1 c1(NC(N2CC(F)(C(=O)Nc3c(C(=O)OC)ccs3)C2)=O)cccc(Cl)c1Cl N1(CC#C)CCCN(S(=O)(=O)C2CC(C(=O)NC3CC3)C2)CC1 C(C(CC(C)C)NC(c1csnc1Br)=O)NC(C1(COCC)CC1)=O C(=O)(CCCC(=O)NC(CN(C(=O)C(CCC)c1ccccc1)C)C)OCC C1(CC(=O)NCC2CN(C(=O)C3CC3)CC(C)(C)C2)(OC)CC2(CCOCC2)C1 CC(C)CCC(O)C(=O)N1CCN(C(=O)CCc2cnn(C)c2)CC2(CC2)C1 c1(OCC(=O)NC(CN(C(=O)CCCC#N)CC)C)c(C)nn(C)c1C C(Cc1ccccc1)(CCNC(=O)Cc1cncn1C)NC(CC=CCC)=O Cc1nc(N2CCC(NC(=O)CC3COCCO3)C(C)C2)cc(Cl)n1 C1(COC)(CNC(C2CCN2C)=O)CCCN1c1nnc(-c2ccon2)s1 Cc1ccccc1-c1cn(CC(C2CC2)NC(=O)CCN2CCCC2)nn1 CC(CCC(C)(C)C)C(=O)NC1(C(=O)NC2CCn3cncc3C2)CC(F)C1 N1(C(CN(C2CCSC2)C)=O)CCCC(C2CCN(C(=O)C(C)(C)CC3CC3)C2)C1 Cn1nc(Br)c2ccc(C(N3C4CN(C(c5ccc(I)cc5)=O)CC34)=O)cc12 N1(C(c2c(C)c(Cl)cnc2)=O)CC2CN(C(=O)CSC(F)F)CC2(C)C1 Cn1ccc2ccc(C(N3CCCC3CNCc3cncc(Br)c3)=O)cc12 C1(C(=O)NC2C(F)CCN(C(CCCC)=O)C2)CCc2nc(C3CC3)ncc2C1 CCC(CNC(C1(F)CCN(C(=O)C(O)CC2CCCC2)CC1)=O)C(C)(F)F C(=O)(CCCCCO)N(CC(CN(C(C)=O)C)O)C c1(CNC(C2CCCN2C(N)=O)=O)ccc(CN)c(F)c1.N1(C(N)=O)CCCC1 C#CCC(C)C(=O)N1CCCC(N(C(=O)CCc2cnoc2)CCF)C1 C1(NC(=O)C=CC2CCOC2)CCCN(C(=O)CCc2ccco2)CCC1 C(CCCC(C)(C)C(=O)NNC(=O)C1CCCCCC1)NC(C(C)C(C)(C)C)=O c1(C(N(C2CC2)CC2N(C(COCCC)=O)CCC2)=O)cnc(O)n(C)c1=O C1(NC(C(CC)(C)C)=O)CC(F)(F)CC1NCC1CCN(C(C)=O)CC1 C1(NC(c2noc(C3CC(OCC)CCO3)n2)CC)CC(O)C(O)C1 N1(C(C(CCC)N(C)C)=O)CC2CC(C1)N(C(c1nn(CC)nc1C)=O)C2 N1(N(C)C)CCN(C(=O)CCC2(C=O)CC2)CC1C(F)F c1(C(=O)NCCNC(=O)CO)cc(N2CCCC(COC)C2)ncn1 O=S1(=O)CC(NCC2CC(O)(c3ccccn3)C2)C2CCCCN12 c1(OC)cccc(O)c1C(N1CCN(C(c2cc(C)c(C)o2)=O)C(C(F)F)C1)=O Cc1cc(O)cc(Cl)c1C(=O)NC1CCCCC1CNC(=O)CCCN(C)C N1(C(CCOCC)=O)CC(NC(c2cnc(N(C)C)s2)=O)CC(C)C1 c1(OC)cc(F)ccc1C(N1CCN(C(=O)C(C)(C)C2CCOCC2)CC1C)=O C(=O)(C(F)CC(C)(C)C)NC1CC(CCNC(c2c(C)n(C)nn2)=O)C1 Cc1nnc2ccc(C(N3CCCC(CO)(NC(C45CCCC4C5)=O)C3)=O)cn12 CC1CNCC(CC(=O)NC2CCN2C(=O)CC(c2ccc(Cl)cc2)O)O1 CCCCCC(C)(CC)C(=O)N1CC2(CC(NC(=O)CC3CC=CCC3)C2)C1 C1(C(=O)NCCCC2N(C(c3c(CC)c[nH]c3)=O)CCC2)C2CC3C(C2)C13 C1(NC(c2nccc(OC)c2OC)=O)C(C)CN(C(c2cnc(Cl)[nH]2)=O)CC1C CS(=O)(=O)c1ccc(F)c(C(=O)NCCCSCc2cccnc2)c1F N1(C(CC2(C)CC2(F)F)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)CC12CCC2 c1(C(C(N2CC(CC(C)NC(C(F)=CCC)=O)C2)=O)O)ccc(O)c([N+](=O)[O-])c1 c1(C(N2CCC(NC(CCNC(=O)OC)=O)C2)=O)ccc(C(C)(F)F)cn1 c1(C(CCC)C)nc(-c2ccc(C3CCC(=O)N3)cc2)n(-c2cccnc2C)n1 C(=O)(C1c2ccccc2C1)NC(COC(C)C)C(=O)NC1CCCN(C)C1=O c1(OC)ccc(Cl)c(C(=O)NCC(C)CNC(c2nc(C)ccc2C)=O)c1F n1(C(C)C)ncc2c(NCC(F)CO)[nH]c(=NC3CCCCC3F)nc12 N1(C(CCSC)=O)CCc2c(c(CNC(=O)C(C3(O)CCCC3)F)nn2C)C1 C1(C(=O)NCCC2(O)CCN(C(CNC(C)=O)=O)C2)CCc2nnc(O)n2C1 c1(C(N2CCN(C(c3ccc(C)nc3)=O)C3C2C3)=O)ccc2occc2c1O c1(C(N2CC(C(C)NC(C3CC(C(F)F)C3)=O)C2)=O)cccn2nncc12 C(=O)(CC1CC(C(C)C)c2ccccc21)N1CCC(NC(CCC#C)=O)C(O)C1 c1(CNC(c2ccc(Cl)cc2Cl)=O)ccc2nc(N3CCOCC3)[nH]c2c1 Nc1ccc2nc(N3CCCC(CO)(NC(=O)C=Cc4ccccn4)C3)sc2c1 c1(C(=O)NCC2(CNC(CSCC(C)C)=O)CC(F)(F)C2)cc(S(N)(=O)=O)c[nH]1 N1(C(C(CCSC)OC)=O)CCC(N(C(=O)C=CC(=O)OC)C)C2(CCC2)C1 C(=O)(C(C)CC(F)F)NC(C(=O)NCc1ccc(C)cc1)C1CCC1 N(C1COc2cc(F)c(Br)cc21)C(C1C(C(C)(C)C)CC1)=O c1(OC)ccc(C(=O)NC2CN(C(C3(C#N)CC(=O)C3)=O)CCC2C)c(C)c1 N1(C(COC(CC)(C)C)=O)CCC(C(C)(C)NC(c2cc(CO)on2)=O)C1 N1(C(c2c(NC)cnnc2)=O)C2CCC1C(C(=O)N(C1CC1(F)F)C(C)C)C2 CCCCC(C(N)=O)NC(=O)CCNC(=O)COC1CN(C(C)=O)C1 c1(C(N2CC(C(=O)Nc3c(C)c(Br)c(Cl)nc3)C2)=O)c(F)ccc2[nH]ccc12 c1(C(=O)NCC(CNC(C(C)(C)c2ccno2)=O)F)cnc2n1CCS2 N1(C(CC=C(C)C)=O)CCC(NC(c2nccc3nn[nH]c23)=O)CC(C)(C)C1 C1(NC(C(COC)(C)C)=O)COCC1C1CC1.c12nscc1C(=O)N2 CC(C)(CC(=O)N1CC(F)(F)CC1CNC(C1C2CC3C(C2)C13)=O)C(F)F c1(C(N(CC(CNC(C2C(C(C)C)OCC2)=O)O)C)=O)cnc2c[nH]nc2c1 c1(C(=O)NC2CN(C(=O)C=C3CCC3)C2)cc2sc(N3CCCC3)nc2s1 C12(C(=O)NCCOC(CNC(C(c3ccn(C)n3)C)=O)(C)C)CCC(CC1O)C2 Cc1[nH]c2ccccc2c1CC(=O)NCC(F)CNC(=O)Cc1cc[nH]c(=N)c1 S(=O)(=O)(c1cnc(N(C)CC2CC2)c(Cl)c1)N(C)Cc1cc2ccccc2s1 c1(CNC(CC2C(CNC(CC(CC)C)=O)C2)=O)cc(C)nc(C)c1 CN1CC(C(=O)NC2CC(NC(C3CC(=O)N(c4nccs4)C3)=O)C2)CC1=O C1(NC(c2c(CC)ccs2)=O)CN(C(=O)C(O)CC(F)F)Cc2ccnn2C1 N1(C(C)=O)CC(C)(C)OCC1C(C(=O)CS(=O)(=O)NCC1CC1)=O.C12CC(C1)N2 c1(NC(=O)Nc2cccc(CO)n2)ccc([N+](=O)[O-])cc1 CC(C(CCc1ccccc1)NC1COCCOC1)NC(=O)OC(C)(C)C c1(Cc2c(C)non2)nc(CO)nn1-c1ccn(C2CCOCC2)n1 Cc1c(Br)c(C(=O)NCC2(O)CCN(C(=O)C3=CC(C)(C)C3)C2)nn1C C(=O)(C1CCCc2ncc(C)n21)NC(C1CCCC1)CNC(CNC(C)=O)=O c1(C(=O)NCC(CNC(=O)Cc2ccsc2Br)OC)c[nH]c(=O)cn1 c12cn(nn1)CC(=O)NC2.c1(CC(COC(F)F)N(C)C)ccccc1 c1(C(=O)NCC2C(NC(c3ncn(CC)c3)=O)C2)ccc(=O)n2c1CCCC2 N1(C(C(C)OCCOC)=O)CCC(CN(C)C(C2(C(N)=O)CCC2)=O)C1 C1(OC(C(C)(C)N(CC(C)(C)C)C)=O)CC2(CCN(C)C2)CO1.C(C)(C)(C)OC(=O)O C1(C(=O)NCCC(C(C)C)NC(c2cnc(N)c(O)c2)=O)Cc2ccccc2O1 Cc1ccc(F)c(C(N2CC(F)CC2C(=O)NC2CC(n3ccnc3)C2)=O)n1 N1(C(C2N(Cc3ccc(OC)cc3C(F)(F)F)CC2)=O)C2CCC1CC(CO)C2 c1(OC)c(C(=O)N(C)CC2CCCN(C(C3(Cl)CC3(C)C)=O)C2)nc(O)nc1O C(=O)(C(C)(C)C1=CCN(C(c2ccc(OC)cc2)=O)C1)N1C(C#C)CCC1 c1(C(=O)OC)ccc(C(=O)CNC(=O)C(C)COc2ccccc2)cc1 C1(OC)CN(C(=O)C(C)(C2CC2)OC)CC1C(N1CC(C#N)(CCF)C1)=O C(=O)(C(C)C(=O)N1CCCC1CN(C)C(c1csc(-c2cnccn2)n1)=O)OC N1(C(c2c(C)nsc2)=O)CC2(C1)CN(C(=O)CCc1ccn(C)c1)CC(C)(C)O2 C(C)(CCCN=c1[nH]cc(C#N)cc1C)NC(C(C)OCC)=O Cc1cc(O)cc(C)c1C(=O)NCC1CCCN(C(=O)C(C)C(C)C)CC1 N1(C(C(C)S(C)(=O)=O)=O)CCC2C(CCCN2C(=O)CCCCN(C)C)C1 C1(CC(C)NC(C(C)NC(C)=O)=O)CCN(C(c2c[nH]c(=O)cn2)=O)CC1 C1(CNC(c2cnc(O)s2)=O)CCCN(C(c2ccccc2C2CCC2)=O)CC1 N1(C(CNC(C(C(C)C)N(C)C)=O)=O)CC(O)CCC1C c1(C(=O)NC2CN(C(C(C(C)C)CN(C)C)=O)C2)noc2c1CC(C)(C)CC2 C(=O)(C(C)(C)C(F)F)NC(C(C(=O)N1CC(CC(=O)OC)C1)C)C C1(C#N)(C(=O)NC2(C(N(C)CCC3CCCO3)=O)CCC2)CCC1 C(=O)(C1=Cc2ccccc2OC1)N1C2CCC(NC(C(N)=O)=O)(CC2)C1 C(CC(=O)NCCn1ccnc1)(C(F)F)N(C)C(c1cc[n+]([O-])cc1)=O C1(CCNC(c2c(-c3ccccc3)noc2C(=O)C2CC2)=O)CCCCC1CO C(=O)(C1=CCC(C)(C)CC1)N1CC(C#C)(C(N2CCC(n3cncn3)C2)=O)C1 n1(CCC)nnnc1C(C1(C(F)(F)F)CCC1)NCCC(C)(O)C1CC1 C1(NC(C2(C#C)CN(C(c3ccc(C(C)C)o3)=O)C2)=O)CCC12CCCC2 C(C(C)(C(C)C)NC(c1nc(Br)c(C)s1)=O)NC(C1(C#C)CC1)=O C1(NC(CC(C)c2ccco2)=O)CCN(C(=O)CN2CCCS2(=O)=O)CC12CC2 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCN(C)CC1CNC(=O)CN1CCC1C C1(C)(C(=O)NC2(CO)CN(C(C3CCC(SCC)CC3)=O)C2)CCC(O)CC1 C1(C(=O)NCc2ncn(C)c2)C2CCN(C(c3cc4n(n3)CCO4)=O)CC12 C1(C(=O)NCCCCCC)C(O)CCN1C(=O)COc1ccccc1 C1(CSCC(=O)NC(C(=O)Nc2cccnc2)C2CC2)CCCCCC1 c1(C(=O)NC2CC(C)(NC(c3cnc(C4CC4)s3)=O)C2)cncc2cccnc12 C1(N(C(c2csnc2C)=O)CC)CCN(C(=O)CC2COCC2O)C1C C1(C(=O)OCC)CC2CCC1CN(C1CCOC(C)(C)C1)C2 Cc1nc(C)c(C(=O)NCc2occc2C(=O)NCC2(O)CCN(C)C2)o1 C(C)(CCCCN=c1nc(-c2ccccc2)[nH]s1)NC(C1C(OC)C1)=O N1(C(C2C3CN(C(c4c(C#C)c[nH]n4)=O)CC32)=O)CCCC[Si](C)(C)C1 CC1CN(C(C2CCN3CCC2C3)=O)CCCN1C(c1ccc(F)c(F)c1)=O CC(C)(CNC(=O)CCc1ccsc1)CNC1(CC(=O)OC(C)(C)C)CC1 C1(C(N2CCCC(CC)(NC(c3csc(=NC)[nH]3)=O)C2)=O)CC2(C1)CC(C)(C)C2 O=C(CS(=O)(=O)c1ccc(C)cc1)NC1CCC(CN=c2[nH]cncc2Cl)C1 N1(C(C2(OCC)CC2)=O)CCCC(C(=O)NC2CC(SC)C2)C1 C(CC1CC1)(C(=O)NCCCN(C)C(C1CC2CC2C1)=O)OC N1(C(c2cc(C)n(C)n2)=O)CC2CC1CN2C(=O)OC(C)(C)C CCCC(C)(C)CC(=O)N1C(CC(=O)Nc2c[nH]ccc2=O)C2CCCC12 C(=O)(C=C1SCC(=O)N1C)NCC1CCCN(C(C2CC(C(=O)OC)C2)=O)C1 N1(C(C2C(OC)CN(C(=O)C(CN(C)C)N(C)C)C2)=O)CCC2(CNC(=O)C2)C1 C1(NC(C2N(C(CCC)=O)CCCC2)=O)CN(C(=O)C(C)=C2CC2)CC1C1CC1 C1(NC(=O)CCc2ccsc2)CCN(CCCNC(c2occc2C2CC2)=O)C1 C(=O)(CC(CC)C(F)F)N1CC(C2C(C(NOCCC(=C)C)=O)C2)C1 c1(C(N2CCC(CNC(CCC)=O)(OC)CC2)=O)cnc2nc(Cl)ccc2c1 c1(C(N(CCCCN(C(=O)CCc2cnn(C)n2)C)C)=O)nc(O)[nH]c(=O)n1 C(=O)(C1CCN(C)c2ccccc21)NCC1C(C)CCN1C(C1CNC(=O)N1)=O C1(NC(Cc2nc(C)[nH]n2)=O)CN(C(C2CCCC(=O)N2)=O)CC1C C=CCCCC(=O)N1CCCC(N2CCN(C(=O)CC(CC)C3CC3)CC2)C1 c1(C(=O)NC2(C3N(C(c4n(CC)ncc4)=O)CCCC3)CC2)cccc(C)c1C Cc1cc(CN(C)CC2CCCN(C(=O)C=Cc3ccsc3)C2)sc1C c1(C(C(N2CCC(NC(=O)C=CCCCC3CC3)C2)=O)=O)ccc(F)cc1 CC1OC2(C(=O)NCCCCCCNC(C3CC4CCC4C3)=O)CC1C2 C1(n2c(CCCC)nc(CCCCO)n2)CCc2nccn2CC1 N1(C(CNS(C)(=O)=O)=O)Cc2ccccc2OC2(C1)CN(C(=O)CNC(N)=O)C2 c1(C(=O)NCC(C)CN(C(=O)C(COc2ccccc2)OC)C)c[nH]c(=O)cn1 c1(C(C)C(=O)NC2(CNC(=O)CCS(C)(=O)=O)CC2)cc2ccccc2s1 C(=O)(CC1OB(O)c2ccccc21)N1CC(NC(C(C)(O)C2CCC2)=O)C1 N1(C(COCC(=C)C)=O)CC2CCC(Nc3cc(C)c(C#N)cn3)C2C1 C(=O)(C1=NN(CC)C(=O)CC1)N1C2CN(C(C3(CC=C)COC3)=O)CC1CC2 C1(CCC(C)C)(CC)CCCN1C(=O)OCC1(C#C)COC1 C12(C(N(CCC(C)NC(C3(CC#C)CC3)=O)C)=O)C3CCC(CC13)C2(F)F c1(CN2CC(SC)C(Cn3cc(C4(N(C)C)CC4)nn3)C2)cc(C)c(F)cc1Br C(=O)(CCCCO)NCC(CNC(C1C(c2cn(C)nc2)CCC1)=O)O C1(C(=O)NC(C(C)C)CNC(=O)C(C)(O)c2ccccc2)CCCCC1(F)F N1(CC(N2CCC3(C2)CN(C(c2cnc(O)o2)=O)C3)=O)CCCCCCC1=O C(C(C)(C)NC)OC(C1(C(N)=O)CC1)=O.C(C(O)C1CC1)N N1(C(Cc2cc(C)no2)=O)CCC(F)(CNC(=O)CC2CCC3CC23)CC1 N1(C(C(CCSC)O)=O)C2CCC(C2)C1CC(=O)NCc1cc(C(N)=O)co1 c1(NC(C=C(C)CNC(=O)CCc2nc(O)n[nH]2)=O)ccsc1C c1(C(=O)NCc2c(CNC(=O)CCF)cccc2)cccc(=S)n1O C1(CNC(CCN2CCN(C)CC2)=O)CCC12CCN(C(=O)CCC#N)CC2 C1(C)(C(=O)NCCOC2CN(C(COCC(=C)C)=O)C2)CC(C#N)C1 N1(CC(=O)O)CCCN(C(c2c(O)cccc2Br)=O)CC1 c1(CNC(=O)Nc2ncc(Cc3ccc(Cl)cc3)s2)ccc(Cl)cc1Cl C1(CC)CN(C(C2(COC)CCC2)=O)CC1C(=O)NC12CSCC1C2 N1(C(C2(NC(c3cnn(C)c3N)=O)CC(F)(F)C2)=O)Cc2ccncc2C1 C(=O)(C(C(C)C)C(C)C)N1CC(C)(OC(CNc2c(C(C)=O)cccc2Cl)=O)C1 N1(C(C2CC(C)(O)C2)=O)CC(c2cn(Cc3ncon3)nn2)C(O)C1 c1(C(N=c2nnn(CC)[nH]2)=O)cc2cnccc2[nH]1 C1(OC)CN(C(=O)C=CC2CCOC2)CCC1NC(c1cccc(OC)c1C)=O CN1CCC(N(C(=O)C(C2CC2)N(C(=O)Cc2ccc(F)cc2)C)C2CC2)C1=O c1(CC)ccc(NC(=O)C(N2CCCC(CNC(C)=O)C2)C2CCCCC2)cc1 c1(C(N2CC(CNC(c3csnn3)=O)C(O)C2)=O)cc(F)cc2cnccc12 C1(N(C(c2cscc2Br)C(=O)NCCC2CC2)C)CCC(C)(C)C1 N1(C(C(CC=C)CC)=O)CCCC(C)(C)C1CNC(c1ccc(F)cc1F)=O c1(C(=O)NCC(CCOC)NC(c2cc(CCC)[nH]n2)=O)ccccc1SC c1(NCC2CC(OC)(OC)C2)ncc(C)cc1S(=O)(=O)Nc1cc(F)ccc1C c1(SC)ncc(C)c(N2CCN(CC3CCCCC3N(C)C)CC2)n1 C1(C(=O)NCc2c(C)nn[nH]2)CC=CCN1C(C1CC(CC2CC2)C1)=O CCCC(C(=O)OC)C(=O)NCC1CC(F)CN1C(=O)CC1CCC(=O)NC1=O C#CCCC(C(=O)NC1CC(=O)N(C)C1=O)NC(=O)CC1CCCCCC1 C(C1CCOCC1)=CC(=O)N(C(C(=O)N(C1CCN(CC)C1)C)C)C1CC1 CCC(COC)C(=O)N1CC(NC(c2sc(CC(F)(F)F)nc2C)=O)CC1C CCC(C)CC(C(=O)NCCc1cnco1)NC(c1c[nH]cc1C)=O C(=O)(C1Cc2ccccc21)Nc1cccn2ccnc12.CC12CC(O)CN1C2=O CC1CCN(c2ccc(CNC(C3CC(O)C3)=O)cn2)CC1 C1(C(=O)NC(CC)CNC(C2CCC(C)(C)CO2)=O)CCC2(CCCC2)CC1 C(C(C(=O)N(C(C)CNC(c1cc(C2CCCCC2)[nH]n1)=O)C)OC)OC C(=O)(C(C)(F)C(=O)OC)N1C(C(CC)NC(=O)Cn2[nH]c(C)nc2=O)CCC1 C1(C(C(=O)NCCC#N)N(CCOC)C(C)C2CC2)CCC(C)C1 N1(C(C(CC=C)(C)C)=O)Cc2occ(C(N3CC(=O)NC(CC)C3)=O)c2C1 c1(N(C(c2scnc2Br)C(=O)NC)CC)ccccc1Cl.c12ccc(cc1)OC2 c1(CC(N2C(C3CCCN(C(C)=O)C3)CCCC2)=O)sc(OC(C)C)nc1C N1(C(Cc2c(C)noc2C)=O)CCC2(CCCN(C(c3cccnn3)=O)C2)CC1 C1(C(N2CCC(CCO)CC2)C(=O)N)CCCOCC1.C(CCF)N1CCC1 c1(OC)c(C(=O)N(CCN(C(=O)CSCCCl)C)C2CC2)cc(F)cc1F c1(CNC(C2C(C)(C)CC2)=O)nc2ccc(F)cc2s1 c1(OC)ccnc(O)c1C(=O)NC1CCC(N(C)C(c2nccn2C)=O)C1 C1(NC(COCCOCC)=O)CCCCN(C(c2ccc(OC)cc2F)=O)C1 c1(N2CCC(N(C(CCC)=O)C)CC2)nn2cc(C)nc2s1 c1(CNC2C(C(=O)Nc3ccc(O)nc3)CC2)cc([N+](=O)[O-])ccc1Cl C1(NC(c2c(C)n(C)cc2)=O)CCN(C(c2cnc(C3CC3)nc2O)=O)CC1C C1(C(=O)NC(c2cnn(C3CCC3)c2)CC)CC(O)CN1C(c1scnc1Cl)=O N1(C(C=[SH](C)=O)=O)CCCC(O)(CO)C1.c1(C(N(C)CCN)=O)cc(C2CC2)n(C)n1 c1(C(=O)NCC2(F)CCCN(C(c3ccccn3)=O)C2)cc2cc(F)ccc2o1 C1(C(=O)NCC(CC)NC(c2ccccc2F)=O)CCCC(N(C)C)C1 CC1CCC(C(=O)NCC(C)CNC(C2(C#N)CCCO2)=O)CC1C c1(C(N2CCCC(NC(c3ncc(CC)cn3)=O)C2)=O)ccc(C)c(C)c1 N1(C(C2C(C)C2)=O)CCCC2(CCCN2C(=O)C(c2ccc(Cl)cc2)O)C1 N1(C(C)C(F)(F)F)CCC(C)(NC(=O)CC(C)n2cccn2)C1 N1(c2nc(N(CC(=C)C)C)c3c(n2)CCS3)CCc2sc(S(N)(=O)=O)cc2C1 C(=O)(C1=CC2(CCNC2)C1)NC1C(CCCOC)CC1 N1(CC)CCCCC1C(=O)NCC1CC(NC(=O)C2=CCOC2)C1 N1(C(C(OC)OC)=O)CCN(C(C2CN(C(C)=O)C2)=O)C2CCCC12 CC(CNCc1cn(-c2ccccc2)nc1C(C)(C)C)S(N)(=O)=O c1(C(N(CC(O)CN(CC(=O)Nc2ccccc2)C)C)=O)ccccc1C(C)(C)C c1(C(N2CC(CC=C)(NC(=O)Cc3cnns3)C2)=O)cc(N)cnc1C c1(CC)cnn(C)c1C(=O)NCc1cc(C)c(C(=O)NC2CC23CC(O)C3)o1 C1(C(=O)N(CCCNC(=O)COCC2CCCO2)CCO)(CC)CC(C)(C)C1 c1(N2CCC(N(C)C(c3ccc([N+](=O)[O-])s3)=O)C2)nc(Cl)nc2nc(Cl)n(C)c12 C(=O)(CC(O)CCCC(F)(F)F)NCCC1CN(C(c2ccc(C#C)cc2)=O)C1 N1(C(C(C)OCC=C)=O)CC(CNC(c2ncn(C(C)C)n2)=O)OC2(CCC2)C1 C1(F)(CNC(C(Br)=C(C)C)=O)CC(NC(=O)CCc2ccccn2)C1 C1(C(N2CC(CC(CNC(c3c(CC)non3)=O)(C)C)C2)=O)CC1C1CC1C c1(C(C)C)ccc(F)c(C(N2CCC3(NC(C45CSCC4C5)=O)CC3C2)=O)c1 N1(C(C(C(C)C)OC)=O)CCCN(C(c2ccc(C(F)(F)F)c(F)c2)=O)CCC1 c1(C(c2nnnn2CC2CC2)(C)NC2CC(C(N)=O)C2)cccc2ccsc12 c1(C(=O)OC)c[nH][nH]c1=NC(=O)C1(c2cc(C)c(-c3ccc(OC)cc3)cn2)CC1 C1(C(c2nnnn2C2CCOC2)NCc2nc(C)c(C)o2)(OC)CCCCCC1 C1(C(NOCCN(C)C)=O)C(C2CC2)CCN1C(C12CCC(CC1)CC2)=O C1(C(=O)NCCC2OCCN(C(c3c(COC)ncs3)=O)C2)CCCCC1(F)F C1(NC(CCCSC)=O)CCC(C)(CNC(c2c[nH]nc2C(C)(C)C)=O)C1 c1(C(N2CCCC(C(=O)NCCC#C)C2)=O)nc2ccccc2nc1C c1(C(N2CCC(C3N(C(CC(C)C4CC4)=O)CCC3)C2)=O)cc(Br)n(C)c1 C1(CNC(c2ccc(-c3ncon3)cc2)=O)CCCN(C(C2CCCOC2)=O)C1 c1(C(N2CC(NC(c3c(C)ccnc3)=O)C(CO)CC2)=O)cc(C)c(Cl)c(C)c1 c1(C(=O)NC2C(CNC(C(C)=CC3CC3)=O)CCC2)c(C)nc2sc(C)cn12 C1(NC(c2cccnc2-n2nccn2)=O)CCN(C(c2nc(Br)cs2)=O)CC1F c1(C(=O)NCC2CC(NC(C3(C#C)CCC3)=O)C2)cc(N)cc(C(F)(F)F)c1F N1(C(CCCCCN(C(=O)CCC2CC2)C)=O)CCC2(CNC(=O)N2)C1 C1(CN(CCNC2CC2)CC)Cc2ccccc2O1 N1(C(C(Cn2cncn2)NC(c2cccc(C)c2)=O)=O)Cc2cccc(C)c2C1 Cc1nc2ccccc2n(COCc2ccc(N3CC(C)OC(C)C3)c(F)c2)c1=O C(CC(C)(C)C)(C(=O)NCCC(C)NC(=O)C(c1cn(C)nc1C)C)OC C12(CNC(C(N3CCCC(O)C3)C)=O)CC3CC(C1)CC(C(F)(F)F)(C3)C2 C1(COCC#C)CN(C(C2(C)CCCN2C(=O)CCNC(=O)CO)=O)CCO1 Cc1[nH]c(C(=O)NCCC2CCCCC2C)c(C)c1C(=O)Nc1sccc1Cl N1(C(C2N(C(c3c(CC)[nH]cc3)=O)CCCCCC2)=O)CC(CO)C(C2CC2)C1 Cc1ccnnc1C(N1CCC(CNC(c2c[nH]c(C(F)(F)F)c2)=O)C1)=O Cc1cccc2c(C(=O)N(CCOC)Cc3ccccc3)cccc12 N1(C(C2CCC(C(C)(C)C)C2)=O)CCC(CNC(=O)C(C2(O)CCCC2)=O)CC1 c1(C(=O)NCCCC(C)NC(CCC#C)=O)coc2c1CS(=O)(=O)C2 N1(C(Cc2ccn(C(C)C)n2)=O)CCC(C)(NC(C2CCC(C)CC2)=O)C1 CC(CC(=O)NCCCN(CCO)C(c1coc(C(F)F)n1)=O)c1ccco1 Cc1cc(C)n2nc(CC(N3CCC(N(C)C(c4c[nH]c(Br)c4)=O)C3)=O)nc2n1 N1(C(C)=O)CCCN(C(C2C(NC(=O)CCSCC(C)C)CCC2)=O)CC1 c1(N(C)Cc2ccc(Br)s2)nc2c(c(=NC(C)c3nc[nH]n3)[nH]1)SCC2 C(=O)(C(CCS(C)=O)N(C)C)NC(CNC(c1c(C)nc(C)[nH]1)=O)C(C)C C(=O)(CC(C)CC(C)C)NC1CCCC(N(C(C=Cc2c(C)cncc2)=O)C)C1 C1(N(C(=O)C=CCO)C)CC12CCC(NC(=O)CN1CCN(C3CC3)C1=O)CC2 c1(C(=O)NCC(CC)NC(=O)C(C)(C)N(C)C)ccc(O)c(F)c1 C1(COC)C(N=c2ncnc(COC)[nH]2)CC1(C)C CCCCC(CC(=O)NCCCCCF)NC(c1ncccc1F)=O c1(OC)ncccc1C(N1CCC(C(C)(C)NC(=O)CN2CC(=O)NC2=O)C1)=O c1(C(=O)NCCCCCNC(c2c(C(C)C)cccc2)=O)ccc2c(c1)OCO2 N1(C(c2n(C)ccc2)=O)CC(NC(c2cc(C3CC3)ccc2Cl)=O)CC(C)(C)C1 N1(C(C2(C(C)=O)CC2)=O)CCN(C(=O)CCC2CCCCO2)CC1C C(=O)(CCCC(=O)OCc1cn(C)nc1C(F)(F)F)NC(C)CCCCC(=O)O c1(C(=O)NCC(C)CNC(c2ccncc2N=[N+]=[N-])=O)nc2n(c1Cl)CCCC2 c1(NC(CCc2ccc(OC)nc2)=O)cc2[nH]ncc2cc1OC C1(OC)CCC2(C(=O)NCC34CC(CN3C(=O)CC=Cc3ccccc3)C4)CC12 C1(C(N(CCNC(c2ccsc2Cl)=O)C2CC2)=O)COCCC1c1ccccc1 c1(C(=O)NCC2CC(O)CN2C(C2CC2C2CC2)=O)ccc(Cl)c2ccccc12 c1(C(N(C)CC2(NC(C=C(C)C(C)C)=O)CC2)=O)cn(CC2CCCO2)nn1 c1(C(C)=O)ccc(Br)cc1C(=O)NC(CCC(C)C)c1cccs1 C1(NC(c2ccc(C(C)C)s2)=O)CN(C(c2cnc(C(F)F)s2)=O)CCC1C C=CCC(CNC(=O)CCC(C)N(C)C)C(=O)NC1C2CCCOC12 C1(C(=O)NC2CCCN(C(C(C(=O)OC)C)=O)C2C)CCC2(CC1)CC(O)C2 c1(C(c2nnnn2CC2CCCCCC2)NCC(Cl)C2CCC2)ccccc1F c1(C(N2C(CC(N3CC(CC)OCC3)=O)CC2)=O)cc(C)cc(O)c1 C1(CNC(=O)C(CO)c2ccccc2)CC2CCC(C1)N2C(=O)Cc1cnoc1 C1(Nc2ccc(COCSc3ccccc3)cc2)C2Cc3ccccc3C12 C1(C(N(CCCCN(C)C(C2OCCO2)=O)C)=O)COCC(C)(C)O1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CC(NC(C2(Br)CC2)=O)CC2(CCC2)C1 c1(CCNC(=O)NCc2ccc(C)cc2)cccc(Br)c1Cl CCCC(C)(C)CC(=O)NC1(CC(=O)NCC(c2ccccn2)O)CCC1 N1(C(CCC2CC(C)C2)=O)CCCC(CCCCNC(C2COC(=O)N2)=O)C1 C1(CC)CCCN(C(c2ccc(C)[nH]2)=O)C1C(=O)NCCC(C)N1CCCC1 c1(C(=O)NC2CC(NC(C3(CO)CC3)=O)C23CCC3)cnc2c(F)cccc2c1 C(C(C(=O)NCCNC(N)=O)NC(c1cc(C)c[nH]1)=O)OCC C1(NC(c2onc(C(C)(C)C)n2)=O)CN(C(=O)C(C)(F)F)C2CC12 CC1CN(C(C2(C)CCCO2)=O)CC1CNC(=O)CC1CC2(CC2)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C3=NOC(C)C3)C2)ncnc2c1cnn2C c1(CNC(=O)NC23C(C)(C)C(CC2)CC3)cccc(P(C)(C)=O)c1 Nc1cc(C(=O)NCC2CCC(NC(c3ccc(Cl)cc3Cl)=O)CC2)ncc1F C12(NC(c3cc4c([nH]3)CCCC4)=O)CCCC1CN(C(=O)C=Cc1cscn1)C2 C(C1=NOC2CCCC12)NC(C1CCN(C(c2cncc(Cl)c2)=O)CC1)=O C(=O)(CCCC(=O)N(C1CCN(C(c2cccc(N)n2)=O)C1)C)N(C)C CN1CC(=O)NC(CC(=O)NC2COCCC2NC(=O)C(C)(C)O)C1=O C1(C(=O)NC2CC(OCC)C2)(CO)CCCN1C(C1CCCC(C(=O)OC)C1)=O c1(C(=O)NCC(C)(C2CC2)NC(C(CC(C)C)OC)=O)ccnc2[nH]cnc12 C1(NC(C(C)Sc2ccc(C)cc2)=O)CN(C(c2nc(Cl)sc2Cl)C)CCC1O C1(C(N(CC(C)NC(=O)CCCC2CCOCC2)CC)=O)CC2CC1CO2 N1(Cc2ccc(-c3n(C)cnn3)s2)CC2(CCCC2)c2cccc(F)c21 N1(C(C=C(CC)C)=O)CCC(C2(NC(c3ncn4c3CCCC4)=O)CC2)CC1 C1(C(=O)NCC2(C(N(C)Cc3cn(C)cn3)=O)CC2)CC2(CSC2)C1 N1(C(C2C(C)=C2)=O)CCCCC1C1CCCN(C(c2cc(CO)[nH]n2)=O)C1 N#Cc1cc(F)c(F)cc1NC(C1CCN(C(=O)CN2CCNC(=O)C2)C1)=O Cc1nc(Cl)sc1C(N1CCN(c2noc(C(C)C)n2)CC1)C(=O)NCC1CC1 C(C(O)C(C)(C)C)NC(C(n1cc(-c2cn(CC3CCCN3C)nn2)cn1)C)=O CC(C)CC(C)CC(=O)N(CCC(N1C2CCC1CC(O)C2)=O)C C1(NC(C2CS(=O)(=O)CCO2)=O)CCCC12CN(C(=O)C(F)(F)CC1CC1)C2 c1(C(=O)NCC2CCC(NC(CC(C)C3CC3)=O)C2)cn2cc[nH]c(=O)c2n1 N1(C(c2cnc(OC)nc2)=O)CCN(C(=O)C(C)C(=O)OC)C2CC12 Cc1cc(F)c(C(=O)NC2CCCC(CNC(c3cn(C)nc3O)=O)C2)c(F)c1 C1(N(C(C)C(=O)NCc2ccco2)C)CCCCC1C C1(F)(C(N(C)CC2CCN(C(C3CC(C4CCC4)C3)=O)C2)=O)C(C)(C)C1(C)C C1(C(N2C(c3ccc(C(=O)O)s3)CCC2)=O)CC(CO)C12CCC2 C1(C(N2CC(C)(OC(c3cccc(OC(C)(C)C)c3)=O)C2)=O)CCOC(=O)CC1 C1(CNC(c2c(C)coc2)=O)CCCC2(CN(C(c3cccc(C)c3O)=O)C2)O1 c1(COC)cc(C(=O)NCC=CCNC(C2(F)CC(c3ccccc3)C2)=O)on1 C1(NC(C2C(COC)C2)=O)CC1C1CCCN(C(C2(OC3CCCC3)CC2)=O)C1 N1(c2n(CC=C)c(C(CC)C(C)(F)F)nn2)CC2(C1)OCc1cc(OC)ccc12 c1(C(N(C2CCN(C(C34CCCCC3OCC4)=O)C2)C)=O)ccc(F)c(F)c1F c1(C(=O)NCCC(CC)(CC)NC(=O)C(O)CN(C)C)n[nH]c2c1CSCC2 C1(C2CCOCC2)(C(=O)NCc2cn(C3CCCC3)cn2)CCNC1 CC1CCCC1C(N1CC(C)(O)C1)=O.N12CC(C1)OCC2=O c1(C(=O)NCCC2(C)CCN(C(=O)CC3OCCC3(C)C)C2)cccc(F)c1N C1(O)(CC(=O)N(C(C)CNC(C2OCCO2)=O)CC)CCCCC1 N1(C(C2C(=C)CC2)=O)CCC2(NC(c3cc(Br)co3)=O)CCCC12 C12(C(N3C(C(C)NC(=O)CCC(N)=O)CCC3)=O)CC1COC2(C)C C1(CC(C(=O)C(N)=O)=O)CCN(CCF)CC1.C(C(C)(C)CN)NC C=CC1(C(=O)N(C)CCc2noc(C)n2)CCN(C(c2ccc(F)s2)=O)CC1 N1(C(C(CCC)(C)C)=O)CCOC2(CCCN(C(=O)CNC(N)=O)C2)C1 C1(C(=O)OCC2(CO)COC2)CN(C)CCN1C(=O)Cc1c[nH]nn1.CO Cc1cc(CNC(C2CSC(C(F)(F)F)C2)=O)ncc1[N+](=O)[O-] C12(CNC(C(CC)N(C)C)=O)CCC(CC1)CN2C(=O)CCNC(=O)CO CC1CCCC1(C(=O)NCCCCN1CCC1)NC(=O)CC1CCCC1O CCC(C)C(C)(c1nnnn1C1CCCC1)Nc1cnn(CCC#N)c1C c1(OC)cc(F)c(C(=O)NC(C)C(C)NCc2ccc3c(c2)CCO3)c(Cl)c1 Cc1cc(C(N2CC3CCN(C(c4coc(CO)c4)=O)C3C2)=O)ccc1[N+](=O)[O-] CC1(C)CCOC1C(=O)NC1CN(C(c2ccnnc2)=O)C1 C12(C(=O)NC3(CNC(=O)CCC4CCCCC4)CCCO3)CC3CC1C2C3O c1(NC(N2C(c3nc(C)c(C)[nH]3)CCC2)=O)ccccc1S(=O)(=O)C(F)F CC1CN(C(C2(C)CCCN2C(c2ccc(O)c(F)c2)=O)=O)C(C)CO1 N1(C(C2(C)CC(=C)C2)=O)CCC2CCOCC2C1 c1cc(N2CCCCC2)ccc1NCCC1CCC2CC12 C(=O)(C(O)CCCNC(C1CCC(OC)C1)=O)NCc1c(OC)cccc1 Cc1ccc(C)c(OCCC(=O)NC2C3CC2N(C(c2cc(C)ccn2)=O)C3)c1 c1(C(=O)NC2CN(C(C(COC)COC)=O)CC(F)C2)cc(Cl)cc(C)c1OC C1(CCNC(=O)COC(F)(F)F)CCCN1C(=O)COCc1cc(C(F)F)on1 C#Cc1nccc(N2CCCC(C(=O)NC(c3ccncc3Cl)C)C2)n1 C1(CC(=O)NC(C2CN(C(=O)CC3CC=CC3)C2)C)CC1(C)C c1(OC)cccc(C)c1C(=O)NC1CC1NC(=O)Cn1ccc(Br)n1 N1(C(C(C(C)C)O)=O)CCCC2(NC(c3cc4n(n3)CCCC4)=O)CC2C1 c1(C(N2CC3CC(NC(CC4(C)CCCC4)=O)C3C2)=O)c[nH]c2cc(N)ccc12 C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(CC(=O)NC(COC)C)C1 N1(C(CCCNC(=O)OCC)=O)CC(NC(C2(NC(C)=O)CCC2)=O)CC1C C(=O)(CCCC(C)NC(c1c[nH]c(C#N)c1)=O)NC(C(=O)OC)CO C1(C(=O)Nc2c(C)cccc2)CN(c2nc(C(F)(F)F)ccc2Br)CCC1C Cn1nc2c(c1C(=O)NCCN1CCN(C(C3CCNC3=O)=O)CC1)CCCC2 C1(NC(C=Cc2c(C)ncs2)=O)CCCN(C(=O)CP(C)(C)=O)CC1 C1(C(c2ccccc2)C)CN(C(=O)Cn2cc(C3(C)CCCO3)nn2)CCO1 c1(CC)ccnc(C(N2CCC(F)(C(=O)NCc3nonc3CC)C2)=O)c1 N1(C(C=COCC)=O)CCC(NC(c2ccco2)=O)C(F)C1 c1(C(N2CCN(Cc3ccc(Br)cc3Br)C(CO)C2)=O)cccc2c(Br)n[nH]c12 N1(C(c2scc(OC)c2)=O)CCCC(CN(C)C(c2nnn(C(C)C)c2C)=O)C1 C12(N(CCCC3CCC3)C)CCC(n3cc(Cn4cc(Cl)cn4)nn3)(CC1)C2.OCC N1(C(CONC(C(CSC)C)=O)=O)CC2(CCCCCC2)C1 C1(NC(C2(CC)CCN(C(=O)CCc3ccn(C)n3)C2)=O)CCC2(CCC2)CC1 C1(NC(CCCNC(C)=O)=O)CC12CC(NC(c1cc(C3CC3)ccn1)=O)C2 c1(C(N(CC(C)N(C(C2C(CCOC)C2)=O)C)C)=O)ccc(O)nn1 C12(CNC(CCSCC)=O)CC3CC(CC(NC(=O)C=CC4CCOC4)(C3)C1)C2 C1(F)(C(=O)NCCCCOC(C)C)CCCN(C(C2CC(n3cnnc3)C2)=O)C1 C1(NC(CCN(C2CCCCCC2)C)=O)CCN(C(C2CCCS2)=O)CC1F C1(OC)(CNC(=O)C(C)SC)CN(C(c2occc2Cl)=O)C1 Cc1cccc(O)c1C(=O)NC1CCCC(NC(C2(C)COCCO2)=O)C1 C(C(C)(CO)OC)NC(CN(C(=O)CCc1cn[nH]c1)CC#C)=O c1(-c2n(-c3cccc(Cl)c3)nc(C3CCC3)n2)ccc2c(c1)COC2 C1(NC(N2CCC(OCCN(CC)CC)C2)=O)CCCOC12CCC2 C1(NC(=O)CC2CCOC2=O)C2CC1CN(C(=O)Cc1c(F)cccc1Br)C2 c1(NC(c2cc(O)no2)=O)cncn1C.C12(CCC1)N(CC)C2=O CCC(Cc1ccccc1)CC(=O)N1CCC1CNC(c1ncccc1Cl)=O CC1CCN(C(=O)COC(F)F)CCN1C(C1CCCOC12CCC2)=O C(C(C)(CC)C(=O)Nc1cc(OC)cc(O)c1)NC(C(C=C)OC)=O NC1(C(=O)NC2CC2Cc2ccc(F)cc2)CC12CCC2 Cc1ncccc1C=CC(N1CC=C(CNC(C2CC(C)CO2)=O)CC1)=O c1(CCC(=O)NCC(CC)(C)NC(=O)C(=O)C(C)(C)C)ccc(OC)c(Cl)c1 N1(C(CC2(OC)CN(C(C(C)OCCC=C)=O)C2)=O)CC(C(N)=O)C(C2CC2)C1 C1(C)(CC(C)C)CCCN1C(C1C2CC1N(C(c1coc(C(N)=O)c1)=O)C2)=O n1(CC(N2CCCC(OC(F)F)C2)=O)c(-c2ccccc2)nc2ccccc12 c1(OC)noc(C)c1C(=O)NCCC1(C(=O)NOCC2CCCO2)CC1 N1(C(COc2c(C)cc(Cl)cc2)=O)CCC2CCCC12CNC(=O)C(O)C1CC1 CC(=O)CCCC(=O)N1CCC(N(C)C(c2ccc(-c3cscn3)nc2)=O)C1 c1(NC(N2C(CC)CC2)=O)ccc(C)nc1 C(CCCC(=O)NCC1CCOC1C(=O)NC1CC(=CCN2CCC2)C1)OC CC1CCN(CC(=O)N(C(C)CN(C)C(c2ccn(CCF)n2)=O)C)CC1 c1(C(=O)NCC)ccncc1NC(=O)NC1CC(C)CCS1 c1(CNC(C2C(C)(C)COCC2)=O)cccc2c1CCC2 C12CCC(=O)N1C(=O)N(CC)CC(C)NC2=O.c1(SC)csc(-c2cnc[nH]2)n1 C(CCN(C(=O)C=CBr)C)(C(C)C)NC(C(CC)OC1CCCC1)=O c1(C(N(C(C)C)C)=O)ccc(C(=O)NC2(C)CN(c3ccc(Cl)cc3)C2)cn1 C1(N(C(=O)Cc2cnccn2)C)CN(C(c2cn(C)c(C(F)F)n2)=O)CC12CC2 CCC(C)CCC(=O)N1CCC(Cn2cc(-c3cccc(OC)c3)nn2)C1 C(=O)(C(O)C1=CCCCC1)NCCCCCNC(c1nn(CC)c(O)c1)=O c1(OC(C)C)cc(CNC(N2CCC(C)(c3cccc(Cl)c3)C2)=O)cc(F)c1 c1(OC)cc(OC)c(C(=O)NCCCCN(C)C(c2cocc2C)=O)cc1OC c1(NCC(CN(C)CC)(C)C)ccc(OCOC)c(-c2cscc2C(N)=O)c1 C1(CC)CN(C(=O)Cn2cnc(C(=O)OC)c2)CCC1NC(=O)CSc1ncc[nH]1 c1(C(N(CCNC(=O)C(F)C2CCC2)CCOCCO)=O)ncc(Cl)nc1Cl C1(CC(=O)NCCN(CCC)C(c2cn(C(C)C)nc2C)=O)CC(C)(C)CO1 N1(C(C2C(C)(C)OCC2)=O)CCCC(O)(CNC(C2CN(CC)C2)=O)C1 c1(C(=O)NCCN2CCOCC2C2CCCC2)cc2nc(F)ccc2o1 N1(C(C2(COCC)CC2)=O)CCN(C(=O)C2=NOCC2)C(c2ccnn2C)C1 C1(CC)CCN(C(=O)CS(C)(=O)=O)C1C(=O)NC(C)CC1CC1 CCC(C)C(O)C(=O)NC(C)CC1CN(C(c2csc(-c3ccccn3)n2)=O)C1 C1(C(N2C(CNC(C(CC#C)C)=O)CC(F)(F)C2)=O)CC2(C1)CC(C#N)C2 Cc1ccc(-c2cc(C(N3CC(NC(=O)C(C)Cn4cccn4)C3)=O)n[nH]2)s1 C=C(CNC(=O)CCn1cccn1)CCNC(=O)C(C)(F)c1ccccc1 C1(C(N2C(C=CC(N3C(COC)C=CC3)=O)CCC2)=O)CC(=O)CC(=O)N1 c1(C(=O)NC2(CO)CCN(C(C(CC)N(C)C)=O)C2)cnn2ccc(C)nc12 c1(C2C(NC(=O)NCc3cc(-c4ccoc4)[nH]n3)C2)ccc(Br)cc1 Cc1cc(CN(NC2=NCCC2)CC2CCCO2)c(C)o1 N1(C(C(CC2CCCC2)NC(c2cc(C(C)C)no2)=O)=O)CCC2(CSC2)C1 CP(C)(=O)C1CCCCC1C(N1CC(NC(=O)CC2C=CCCC2)C1)=O N1(C(CN2C(C)CCC2)=O)CC2(C1)CN(C(c1nnn(C)n1)=O)CC2CO N1(C(C(C2CN(C(C3CC3C(C)C)=O)C2)OC)=O)CCCC2(CCC2)C1 N1(C(c2c(C)nco2)=O)CCC(C)C(CNC(=O)CSc2ccc(F)cc2)C1 c1(C(=O)NC2CC(NC(C3C(C=C)OCC3)=O)C2)cc(C)c(F)cc1Br c1(CN(CC)CC)coc2ccc(OC)cc1C=CC(OC)=CC1=CC=NC21.S(C)CCC N1(C(COCCN(C)C)=O)CCCC1C1CCCN1C(=O)C=C1CCCCC1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)NCCCOC1C(C)CCCC1C c1(C(=O)NCC2CC(O)(CNC(C3C4CCC34)=O)C2)ccc([N+](=O)[O-])c(CO)c1 S1(=O)(=O)c2ccccc2CN1.C(=O)(C(C)(N)Cc1ccccc1)N(C)CC C(CCCCCC(=O)N(CC(O)CNC(C12CC1CNC2=O)=O)C)SC S(=O)(=O)(c1cnc(N2CCC(N(C)C)C2)cc1C)NC(CCC=C)(C)C CN1CCC(NC(=O)C(CC(F)F)N(C)C(c2coc(C(F)F)c2)=O)C(C#N)C1 CC1(C)Cc2ccc(C(N3CCC4(CCCN4C(=O)CS(C)(=O)=O)C3)=O)cc2O1 C1(C(=O)NC(C)CC(=O)NC2CC3CCC2C3)COCCC1(F)F N1(C(c2n(C)c(Cl)cn2)=O)CCC2(CCCC2NC(c2cnco2)=O)C1 C(=O)(C(C(C)(C)C)C1CCCO1)NC1(CO)CN(c2cc(COC)ncn2)C1 C1(C(N(C)CCC2CCOC2)=O)CCCCN1C(=O)CCC(=O)N1CCCC1 c1(OC)cccc2cc(C(=O)NC(C)C(C(C)C)NC(c3coc(C)c3)=O)oc12 C1(CNC2(NC(C3CN(C(=O)OC(C)(C)C)C3)=O)CCC2)CC(=O)N(C)C1 N1(C(c2ncn(CC)c2)=O)CCN(C(=O)CCSc2c(C)noc2C)C(C)C1 c1(N2CCN(C(=O)OCC)CC2)ccc(NCCc2cccc(F)n2)cc1C C1(C(N2C(CNC(C3COCCO3)=O)CC(C)(C)C2)=O)CCc2nc[nH]c2C1 C(CCCCC(=O)N1CCCCC1C1CCC1)NC(C1CCN(CC)C1)=O c1(C(=O)OCC)cccc2nc(C(=O)NC3(CO)COCC34CCC4)[nH]c12 CCC(C)C(O)C(=O)NCCN1CCC(NC(=O)CCCn2cccn2)CC1 Cc1cc(C(N2CCC(C(C)NC(c3cscc3C#N)=O)CC2)=O)cnc1O c1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCCC2C)cncc2ccsc12 c1(CCCOC(c2ccc(-c3cccnc3)s2)=O)nc2ccccc2s1 CC1CCN(C)CCN1C(N1CCC(C(O)C(F)(F)F)CC1)=O CCC(C)C(C(=O)N1CCC(OC)C1C)NC(=O)OCC(F)(F)F Cc1cn2cc(C(=O)NCC34CC(CN3C(C3CSCCSC3)=O)C4)nc2s1 N1(C(c2c(CCC)nns2)=O)CC2CC(C1)C(CO)C2NC(c1nonc1N)=O N1(C(=O)Cc2n[nH]cc2C(=O)NC2(CCF)CCC2)Cc2cncnc2C1 c1(CC(=O)NC(CN(C(c2c(CC)occ2C)=O)C)C)cccc2cccnc12 c1(OCCOC)ccc(Nc2cnnc(O)c2S(=O)(=O)NC)c(Cl)c1 N1(C(C(F)=CCC)=O)CCC(NC(=O)COCc2ccccn2)C(CC)C1 c1(C(N2CC(CC)N(C(c3oncc3C)=O)CC2)=O)c(C)ccc(Br)c1F n1(CC(=O)NCC(C(C)C)NC(=O)NC)c(Cc2ccco2)nc2ccccc12 CC(C(=O)NC1CC1CNC(c1cc(C2CC2)nn1C)=O)P(C)(C)=O c1(C(=O)NC(CCOC)C)cccc(S(=O)(=O)CCO)c1 C=CCCCC(C(=O)NC(C)(CO)CC(C)C)NC(=O)CCCOC(C)C C1(CCC(=O)NCC(N(C)C(C2(C)CC2(F)Cl)=O)C2CC2)CCCCN1C C(CN=c1ccnc(C(C)C)[nH]1)(CC(C)C)NC(C1Cn2c(C)nnc2CC1)=O C1(CNC(CCSCC(C)C)=O)CN(C(=O)CC2CCCCC2O)CCCO1 c1(NCCC(C(C)C)c2ccncc2)cc(=NCC(F)CO)[nH]cn1 C1(CNC(C2(CSC)CCC2)=O)C=CC(NC(=O)C(F)(F)c2cnccn2)C1 C(CCC(N)=O)(C(=O)N1CCC(CCNC(C2(C)CC3CC3C2)=O)C1)N(C)C C1(C=O)CCCC2(CCC2)O1.c1(-n2c(C)nc(C)n2)ccc(F)c(Cl)c1 C=CCC(CNC(c1ccc(C2CC2)cc1)=O)C(=O)N1CCCC1(CC)CC C12(CNC(CCC(=O)OC)=O)CCC(CN(C(=O)CCc3ccccc3F)C1)C2 Cn1ccc2[nH]c(C(=O)NC3(C)CCN(C(C4CC=CCC4)=O)C3)cc12 C(=O)(C(C)CC(=O)OC)NCc1scc(C(=O)NC2C(CCOC)CCC2)c1 C1(NC(C2(C3CC3)CC2)=O)CS(=O)(=O)CC1N=c1[nH]ncs1 c1(C(=O)NC2C(CNC(C=CC(CC)C)=O)CC2)cccc([N+](=O)[O-])c1C C(=O)(C1=CC2CCC(C1)C2)N1CC(O)(CCNC(c2cnc(OC)c(C)c2)=O)C1 CC1OCCCC1C(=O)NC12CC(C1)N(C(=O)Cn1ncnn1)C2 c1(C(N2CC(F)(C(=O)Nc3cn(CCC)nc3)C2)=O)cccc(Br)c1 C1(CC=C)(NC(C2(C(C)C)COC2)=O)CCN(C(c2ccc(SCC)cc2)=O)C1 c1(CC)cc(C(=O)NCC2(O)CCN(C(C3(C)CCCC3(F)F)=O)C2)cc(O)n1 C=CCC(CC=C)C(=O)N1CCCC(C(N2CCCC2CC)=O)C1CC C1(NC(c2ccc(C3CC3)cn2)=O)C2CC1N(C(C1(O)CC(CF)C1)=O)C2 C(=O)(CS(=O)(=O)CC(=O)NC1CS(=O)(=O)CC1NC(=O)CSCC(C)C)OC c1(C(=O)NC2C(C)CN(C(C3(CO)CCC3)=O)C2)cc(N)cc(O)c1F c1(C(=O)NCC(C)N(C(CC2(C=C)CCC2)=O)C)cccn2cncc12 C1(N(C)C)CN(C(=O)C=CCC(C)(C)NC(=O)CCc2ccc[nH]2)CC1O N1(C(C(C)(C)C2CCCCO2)=O)CC2CC(C1)CN(C(=O)CC1OCCO1)C2 C1(=O)C(CO)NC(=O)N(C(C)C)CC(C)N1.C1(C(=O)NC(C)(C)C)CC1(F)F C=C=C(C)CC(=O)NCCCC(=O)NCc1cccc(OC)n1 C1(CC(=O)NCCOCCCN(C(=O)C(O)c2cnc[nH]2)C)CCC1(C)C C=C(C)C(C)(O)C(=O)NCC1(CNC(c2cncc(N(C)C)n2)=O)CC1 O(NC(=O)C(c1cccnc1)NC(c1ccn(CCF)n1)=O)CC(C)C N(C)(C1CN(C(=O)C(=O)NC2CC2)CCc2ccccc21)C(CC(CC)OC)=O c1(C(=O)OCCCN(C(=O)Cc2ccccc2F)CC)ccc(NC)cc1 N1(C(C2(SC)CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(O)C3)CC(C)(C)C1 C=CCC(C(=O)N1CCCC1C1(NC(=O)CNC(=O)CNC(=O)OC)CC1)OC CCC(O)CN(C(C1(NC(C)=O)CC1)=O)CC.C12CC(C1)C(=O)NC2 CCN(C(C)c1ccccc1)N(Cc1cnn(C)c1)CC CC1(C)C(c2cccc(Cl)c2)CCN1C(C1CCC(C2CCC2)N1)=O Cc1cc(C(=O)N(C)CCOCCCNC(=O)C(F)(F)c2ncc[nH]2)cc(C)n1 c1(C(=O)NCC2(CO)CCN(C(C3CC=CCO3)=O)C2)ccn2c1CCCC2 S(=O)(=O)(C1CCC(=O)CC1)N1C(C(=O)NCc2cccc(OC)c2F)CC(O)C1 C(=O)(C(C)CC)NC.C1(=O)C(=O)N(C(C)C)CCN(CC)CCN1 CS(=O)(=O)c1cc(CN2CCCC2c2cccs2)co1 CCC(C(=O)OC)C(=O)NCc1nocc1C(N1CCC(CC(C)(C)C)C1)=O c1(CNC(C#CC(=O)N(C)C)=O)c(C)nn2c1CN(C(C1CC1(F)Cl)=O)CC2 C1(C(=O)NC2(CC=C)CN(C(C3(c4ccn(C)n4)CC3)=O)C2)C2CCC(=O)C12 C1(C(=O)NC(CCOC)C(=O)N2CCCC(C(C)O)C2)CCC2(CC1)CC2 C1(CC=C)(N(c2cncn2C)C(=O)CO)CN(C(=O)CC)C1 N1(CCC(=O)NCc2c(C)nccc2)CC2CCC(C1)C2NC(c1cccs1)C CC1CCn2ncc(C(=O)N(C3CCCCN(C(=O)CCF)C3)C)c2C1 c1(CCC(=O)NC(CNC(C2(Cl)C(C)(C)C2)=O)C2CC2)ccc(N)cn1 C(=O)(C(C(C)C)N(C1CC(N(C(=O)CCN2CCCC2=O)C)C1)CC(C)C)OC C(=O)(C(CN=[N+]=[N-])NC(c1occc1C)=O)N(C)Cc1n(CC)cnn1 c1(C(=O)NCC2(F)CCC(NC(C(C)(C)O)=O)C2)cn(CCO)c(=O)nc1O CCCCC(=O)NCC(C)CNC(C1(CCOCC)CCCC1)=O CCC(C)(C)C(O)C(=O)NCC(CC(C)C)C(N1CC2C3C=CC(C3)C2C1)=O c1(CC)cc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCc2cc(C)[nH]n2)n[nH]1 c1(C(=O)NC2CC=CC(n3cc(CNC4CC4)nn3)C2)ccc2nsnc2c1 c1(C(N(CCCNC(C(CCSC)OC)=O)C(C)C)=O)cc(C#N)ccc1N c1(C(=O)NCCN(C(=O)CC2OCCC2C)CC)c(C)sc2ccc(F)cc12 c1(CC(=O)NCC23N(C(c4cnn(C)n4)=O)CC(C2)C3)nn(C)c2ccccc12 C1(CNC(CC2CCN(CCC(C)(C)C)C2)=O)CCC2(CCC2)O1 c1(C(=O)NC2CC(NC(C34CCC3C4)=O)C2)csc(C(F)(F)F)n1 C1(CC)CCOCCN1C(c1scnc1Cl)C(=O)NC(C)C N1(C(=O)C=Cc2ccoc2)CCC2(C1)CN(C(C1CC(CCO)C1)=O)C2 c1(C(=O)NC2CC(C(C)C)OCC2)cc(C#N)ccc1Cl c1(OC)ccc(CCC(=O)N2CCC2NCCc2nn[nH]n2)cc1C(F)(F)F C1(CNC(Cc2c(C)con2)=O)CC12CCN(C(c1cccc(Cl)c1Cl)=O)CC2 c1(C(N2CCC(n3cc(CC(=O)OC)nn3)CC2)=O)cccc2c1CCC2 C(=O)(C(F)(F)c1csc(=N)[nH]1)NCC(CN(C)C(C1(N(C)C)CCC1)=O)O O=C(CCCC1CCCC1)NCC=CCN(C(=O)C=CCN1CCOCC1)C1CC1 c1(C(=O)NC2CN(C(C(CCC)NC(N)=O)=O)CC2(C)C)cncc2c1CCC2 C1(CC)CCC(NC(C2COCCN2C(=O)C=C(C)c2ccco2)=O)CC1 N1(C(c2c(C)noc2C(F)F)=O)CC=C(CNC(c2cc(O)nc(O)c2)=O)CC1 Cc1[nH]nc2ccc(C(N3CC4(CC4)CC3CNC(=O)CC3(C)CC3)=O)cc12 c1(NC(C2CC(=C)CN2C(c2nccnc2OC)=O)=O)cc(Cl)c(Cl)nc1Cl C1(C(=O)NCCOCCNC(c2cc(CCO)on2)=O)CC2COCC(C1)C2 Cc1ccnc(C(N2CC(c3ccccc3)(NC(c3occc3Br)=O)C2)=O)c1 c1(C(=O)NC(CCCNC(c2n(CC)ncc2)=O)C)nc(O)nc(O)c1N C1(O)(CCNC(CCCSC)=O)CCCN(C(=O)Cc2ccc(CO)cc2)C1 c1(OCCC(=O)N(CCN(C(=O)C=CCF)CC)CC)cccc(F)c1 CC1C2CC(C2NC(C2CCN(C)CC2)=O)N1C(=O)C1=CCCOC1 C1(CC)(CO)CCN(C(=O)C(CO)NC(c2ncncc2Cl)=O)C1 C(CNC(=O)C(C)n1ccnc1)(CNC(=O)CC1(NC(C)=O)CC1)OC c1(CC)nc(C#N)cc(=NC(C)CNC(=O)Cc2ccco2)[nH]1 c1(CCCC(=O)NCC(O)CNC(=O)Cc2cnc[nH]2)ccc([N+](=O)[O-])cc1 N1(C(CCCOCC)=O)CCCCC12CC(NC(=O)Cc1ccc(CC)cc1)C2 CC1CC2CCC(C1)N2C(=O)C(CO)NC(c1ccc2cc[nH]c2n1)=O C(=O)(C(C)(O)C(F)(F)F)NCc1oc(C)c(C(=O)NC2CCOC(C)C2)n1 C1(C(N(C(CNC(c2ccc(C#C)o2)=O)C2CC2)C)=O)CC2(C1)CC2(F)F CC(C)(C(=O)NC1CNC(=O)OC1)C1=CCN(C(c2c[nH]c(C(N)=O)c2)=O)C1 C(=O)(C1=C2CCN=C2NC=C1)N1CCN(N2C(CCC3(C)CC3)CCC2)CC1 C1(C(=O)NCCN(C(=O)C2CC2)C(n2cccn2)C2CC2)CCCC1O C1(C(=O)OC)C(C(=O)NCC2(C3CCCCO3)CCC2)C12CC2(F)F C12(C(C)NC(c3ccc(Cl)cc3)CC(=O)O)CC(CCO1)C2 c1(NC(=O)N(C)CCOCCSC)cc(I)ccc1C(=O)CCC(=O)OCC C=CCC(C(=O)N1C(C(N2CC(C#N)C2)=O)CC2CC12)OC c1(C(=O)NCC2N(C(CC(C)C)=O)CC=C2)ccccc1Cc1ccccc1 C(=O)(C(O)P(C)(C)=O)N(CCC1CCN(C(C2N(C)CCC2)=O)CC1)C1CC1 c1(C(=O)NCCC2CC(NC(C3(Cl)CC34CCC4)=O)C2)ncccc1F C1(C(=O)NCc2cccc(CC)c2)CC(C)CN1C(C1CCCC1C)=O N1(C(CC(C)n2cccc2)=O)CCC(O)C(NC(C2CCCN2N=O)=O)C1 c1(C(=O)NC(CNC(C(C)(C)SC)=O)C(C)C)cc(C(F)(F)F)ccc1[N+](=O)[O-] C1(NC(C(C)OCCOC)=O)CN(C(c2ccc(CO)o2)=O)CC1(C)C C(c1nc2ccccc2[nH]1)=CC(=O)NC(C)C(C)NC(c1ccnnc1S)=O C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CC(NC(C(CC)OC)=O)C(F)(F)CC1 c1(OCCOC)ccc(C(=O)NC2CC(NC(=O)C(C)(C)F)C2)cc1OC C1(O)(CN(C(C(CCC)NC(C)=O)=O)C)CCCN(C(C2CC(=O)N2)=O)C1 C=CCC(C)(C)C(=O)NCC1CN(C(c2cnc(O)o2)=O)CCC1C N1(CC(=O)NC2(C)CN(C(c3cc(C(C)C)sn3)=O)C2)CC2C=CC1C2 C(CC1CC1)(C(=O)NCCOC1CCCOC1)NC(C1C(COC)CC1)=O C(=O)(CC1=NNC(=O)C1)NC12C(CN(C(c3c(C(C)(C)C)cc(N)cc3)=O)C1)C2 c1(C(=O)OC)ccc(-n2ccnc2-c2cn(C)nc2SC)c(F)c1 c1(C(N(C)CCOCCNC(=O)CNC(c2ccc[nH]2)=O)=O)ccco1.S(C)C N1(C(c2cc(C(=O)OCC)n(C)c2)=O)CC2CC(C1)C2NC(=O)C(O)C(C)(C)C N1(C(CCC)=O)CC2CCC2(CCNC(C2CC3(CCCC3)C2)=O)C1 C(=O)(C(C)C(C)C)NCCN(C(=O)COc1ccsc1)CC=C Cc1nc(C)c(C(N2CCC(N(C)C(c3ccnc(N4CCCC4)c3)=O)C2)=O)[nH]1 CN1CCN(C(=O)CC2(N(C)C)CCC2)C(CNC(c2cc(C3CC3)ns2)=O)C1 C1(NC(Cn2c(C)nc(C)n2)=O)CC(NC(=O)CN(C)C)C12CCOCC2 Cc1[nH]nc2ncc(C(N3CCC(NC(=O)CC4CCOC4)CC3C)=O)cc12 C1(C(N(C(CNC(c2c(CSCC)cccc2)=O)C)C)=O)CN2CCC1CC2 Cn1cc(C(=O)NC2CC(F)(CNC(c3ccc[n+]([O-])c3)=O)C2)c(C2CC2)n1 c1(C(N2CCSCC2(C)C)C=O)ccc2c(n1)CCC2.c1(NCC)ccccc1Cl CCC(CC(C)C)C(=O)NC(Cc1ccco1)C(N1CC(=O)NC(=O)C1)=O N1(C(C(C(COC)C)C)=O)CCC2(C1)CN(C(c1nc(Cl)ccc1N)=O)C2 N1(C(C2CC3C=CC2C3)=O)CCCC2(C1)CN(C(C1(O)COC1)=O)CCO2 N1(C(c2nc(OCC)sn2)=O)CCC(C)N(C(c2ccn(C(C)C)n2)=O)CC1 C1(CNC(c2n(CCC)nnn2)c2ccnn2COC)CCC(=O)NC1 c1(C(N2CCN(C(c3c(CC)con3)=O)CC2C(C)C)=O)cc2nnn(C)c2s1 C1(F)(CNCc2ccc(C)n2C)CCCN(C(=O)OC(C)(C)C)CC1 C1(N(C)C)CCCN(CCC(=O)NCC2(O)CN(C(=O)CC3CCCOC3)C2)C1 c1(CNC(C(CO)NC(C2C3CC(=O)CC32)=O)=O)ccc(F)c(F)c1 N1(C(C2(C)CCCN(C)C2)=O)CCC2(CC(C(=O)NC(C)(C)C(N)=O)C2)C1 CC(C)C(C)CC(=O)NCC1CN(C(C2CCS(=O)(=O)N2C)=O)C1 N#Cc1ccc(N2CCC(C(=O)NCC3CC(NC(=O)COCCO)C3)C2=O)cc1 c1(C(N2CCCC(C3CCCCO3)C2)C(=O)NC(CC)(C)C)ccc(OC)cc1 c1(OC)c(C)nc(C2CC2)[nH]c1=NCC1(F)CCN(C(c2ccncn2)=O)CC1 c1(C(C(=O)NCCCN(C(=O)CC(C)CN(C)C)CC)(C)O)ccc(F)cc1 C=CCCC(F)(F)C(=O)N1CC(CC(F)C(=O)NCC(C2CC(C)(C)C2)O)C1 C=CCC(C)(C)CC(=O)N1CCN(C(c2c[nH]nc2F)=O)CC(CO)C1 N1(C(c2c(C)cco2)=O)CCCOC(CNC(c2ncccc2C(F)(F)F)=O)C1 C(=O)(CC1=NNC(=O)C1)NC(c1c(OC)cccc1)CNC(=O)Cc1cocn1 c1(CC)ccccc1C(N1CCC1C(=O)NCC=Cc1sccc1C)=O c1(C(N2CC(CCNC(c3nnn(C)c3N)=O)OCC2)=O)ccc2ccnn2c1 C12(CNC(c3[nH]cc(CC)n3)=O)CCCC1CN(C(=O)COCC1CCCC1)C2 C1(CC)CN(C(c2ccc(CNCCCn3cnnc3)nn2)=O)CCO1 CCS(=O)(=O)c1ccc(C(=O)NCC2(CNC(=O)CC(C)CF)CC2)c(N)c1 c1(OC)cc(N)c(Cl)cc1C(N1CC(NC(=O)C(C)(C)CF)CC(O)C1)=O Cn1cc(C(=O)NC2CCC(NC(c3occc3Br)=O)C2)c(-c2cccs2)n1 C(=O)(CCCC(F)(F)C(F)(F)F)NC1CCCCN(C(C=CS(C)=O)=O)C1 Cc1cccc2c(C(N3CC4(CC4)CC3CNC(C3CC3Br)=O)=O)coc12 C(=O)(C(C)C(F)(F)F)NCC1(COC)CCCN1C(=O)CCC=CBr N1(C(C(CSC)OC)=O)CCC2CN(C(C3CC(OC4CCC4)C3)=O)CC12 c1(OC)nccc(CC2(CC(=O)NC(=O)CCSCC3CCCC3)CCC2)n1 N1(C(c2cnc(COC)s2)=O)CCN(C(C2CCCN2C(C)=O)=O)CC2(CC2)C1 C1(NC(C(C)NC(=O)Cc2cccnc2F)=O)CC2(CCC2)C1O Cc1nc(NCCc2cncn2C)cc(=NCc2nc(=N)[nH][nH]2)[nH]1 c1(C(C)(C)C)ncc(C(=O)NCC2CC2NC(=O)CSCC#N)[nH]1 C1(C)(CC)CC(NC(c2[nH]cnc2C)=O)CN1C(=O)COCCCOC N1(c2ccnc(C(N3CCN(CCO)C(=O)C3)=O)n2)C2CCC1CC1(C2)N=N1 C(=O)(CC(C)(C)C(F)(F)F)NCC1CCCN(CC2C(C)OCCC2)C1 N1(C(c2ccc(C(C)C)nc2)=O)CC2CCC1C(NC(=O)C(C)C(C)O)C2 C(CCN=c1nc(O)c2ccccc2[nH]1)NC(=O)CN1Cc2ccccc2C1 C#Cc1ccc(C(N2CC(NC(c3coc(CO)c3)=O)CC3(CC3)C2)=O)cc1F c1(C(=O)NC2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)c[nH]nc1F C1(C(=O)NCC(C)NC(C2(SC)CCC2)=O)CCC(=O)N1Cc1ccccc1F C1(C2CC2)(C(N2CC(N3CCCC3=O)C2)=O)CN(C(C2C3CCCOC23)=O)C1 c1(C(N2C(C(C)NC(CSCCC)=O)CCC2)=O)cc2cccc(OC)c2[nH]1 N1(Cc2n(C)ccc2)CCC2(CCCC2C(=O)Nc2ccc(Br)c(I)c2)C1 CC1CC(NC(=O)C(F)(F)c2ncc(C(F)(F)F)s2)CCO1 C=C1CC(C(=O)NC(c2ccccc2)COC)N(C)C1.S(=O)(=O)(CC1CC1)NC S(=O)(=O)(C1CC2(CC2)C1C(C)C)NCc1c(C)n[nH]c1 c1(CC(=O)N(CC(C)NC(c2cc(C)oc2C)=O)C)ccc(O)c(C)c1 C12(C(N3CCC(COC)C3)=O)CC(CO)(CN1C(=O)C(C)c1cc[nH]n1)C2 c1(C(=O)NCC(CCOC)NC(=O)C(F)(F)C(F)F)cncc(S(C)(=O)=O)c1 CCC(CC)C(C(=O)NC1CCC(NC(c2cnoc2CC(C)C)=O)C1)OC c1(CC)cncc(C(=O)NC2CC(C)N(C(=O)C3=CCCC3)C2)c1 N1(Cc2nc(C(C)(C)C)on2)CCN(CC2CCC(F)(F)C2)CC1 N1(C(CC)=O)CCN(C(C2CCC23CCC3)=O)CC1c1cccc(Cl)c1 C1(C(N2CC3C(NC(c4c(CC)ncnc4)=O)C3C2)=O)CCC2CC(C)CN2C1 C=CCC(CC)C(=O)NC1C=CCCC1C(=O)NCC Cc1ccc(C)n1CC(N1CC=CCC1C(=O)NC1(C2CCCO2)CC1)=O c1(C(=O)NC2(C(F)F)CC(NC(Cc3ccc(C)s3)=O)C2)ncccc1F c1(CC2(C(=O)O)CC2)ccc(F)cc1Cl.c1(C(C(=O)CCN)C)ccccc1 CC(N(C)N1CCC2NC(=O)CCC2C1)C1CC2(CCC2)C1 C12CC(O)CN1C2=O.C1(CNC(C2C(C(=O)OC)C2)=O)CC(F)(CO)C1.C(C)(=O)N C1(NC(c2cc(SCC)ncc2)=O)CCC2CC1CN2C(C1COC1)=O c1(C(N(C)CCNC(=O)CN2C(=O)CN(C)C2=O)=O)cc2c(nn1)CCC2 N1(C(c2c(C)nsc2N)=O)C2CCC1CN(C(=O)CC(C)c1ccncc1)CC2 c1(C(=O)NC(c2cn(-c3ccc(C)cn3)nn2)CCC)cc(C)nc2[nH]cnc12 Cc1ccc(F)c(S(=O)(=O)N2CC3(CC(Nc4ncnc5[nH]ccc45)C3)C2)c1 N1(C(=O)OC(C)(C)C)CCC(C(F)C(C)(C)C)C1.C123CC(C1)(C2)NC3 c1(NC(=O)NCC2(NC(C3CC(N(C)C)C3)=O)CCOCC2)ccc(C#N)cc1 N1(C(Cc2c(C#C)cccc2)=O)CCC2CCN(C(=O)CC(C)(C)OC)CC2C1 C1(CNC(Cc2nnc(C)o2)=O)CN(C(C2CCCC(=O)N2)=O)C2(CCC2)C1 c1(C(N2CC(C(N(CC(C)C)CCC)=O)OCC2)=O)nc(OC)ccc1OC CC(CC(N)=O)C(=O)NC1(CNC(c2cccc(CC(F)(F)F)c2)=O)CCOC1 CC(C)(C)C#CC(=O)N(CC(CC1CC1)C(=O)N1CCC1)CC(N)=O Cc1nc(C(N2CCN(C(=O)Cc3ccsn3)C(CCO)C2)=O)ccc1[N+](=O)[O-] C1(CNC(=O)NC(CSCC)C)CS(=O)(=O)C1 C1(NC(C2N(C(C)=O)CSC2)=O)CN(C(c2cn(C)cc2C)=O)CC12CC2 N1(C(=O)Cc2cn(-c3cnnc(O)c3Br)nn2)CCC2(CCCN(CCO)C2)C1 N1(C(c2ccc(CNC(CS(CC)=O)=O)o2)=O)CCC2CCN(C)CC12 C1(C)(C(N(CC(C)C)CC#C)=O)CN(C(C2C3CCC(F)C23)=O)C(C)(C)C1 C1(CNC(C2(COC)CC2)=O)C(C)CCN1C(c1cc(C(F)(F)F)n(CC)n1)=O C12(C(N3CC4C(N(C)C)C4C3)=O)CC(CN(C(c3cc(F)ccc3F)=O)C1)C2 N1(C(c2cn(CC)nn2)=O)CCC(C)(C)C(NC(=O)CC2CCCCO2)C1 Nc1ccc(C(=O)NCC(C2CC2)NC(c2cc(Cl)ccn2)=O)nc1 N1(C(C=C(C)Cl)=O)CC2CCCC(C1)N2C(c1nc(C)sc1Br)=O c1(CN(C(c2cccs2)CN2CCC2)C(=O)CO)cc2occc2s1 c1(C(=O)NC2CN(C(CC)CC)C(=O)C2)coc(S(=O)(=O)N2CCCCC2)c1 CC(C(=O)N1CC2CC(NC(C3CCC(C)CC3)=O)CC1C2)C(C)C(C)(C)C Cc1noc(C)c1CCC(=O)NC(C)(CNC(=O)C(O)Cc1cccs1)CO C(=O)(C(CCF)NC(c1ccc(O)nc1)=O)N1CCC(COC(C)=O)C1 N1(CC)C(=O)CCC1C(N1CC(F)(CNC(c2scnc2C(C)C)=O)C1)=O N1(C(C(CCSC)OC)=O)CCC2C(C1)NC(=O)CN2C(c1ccc[n+]([O-])c1)=O S(=O)(=O)(c1cccc(=NCc2cc3c(s2)CCCC3)[nH]1)NC(C1CCC(F)(F)CC1)=O c1(C(NC(=NC)NCc2cc(C(F)(F)F)co2)C)cccc(C)n1 C1(CN(C)CC2CCN(C)C2=O)CC2CCC1(NC(=O)C(C)(C)CSC1CC1)C2 N1(C(c2cnc(C)n2C(F)F)=O)CCC(NC(=O)C(O)c2ccco2)C(O)C1 CC1CC(=O)NCCN1C(C(=O)NCCCF)c1ccoc1 CC1CCC(N2CCCC2)CN1C(=O)NCCSCC(c1ccc(O)cc1)O c1(C(=O)NC(c2ccc(NC)cc2)CNC(C(CC)OC)=O)ccc(C#N)cc1 c1(C(N2CC(OC)(CNC(=O)C(C)CF)C2)=O)c(F)ccc(F)c1O N1(C(CN(C(C2(c3nccs3)CC2)=O)CC)=O)CC(C(N)=O)C(C2CC2)C1 c1(C(=O)NC2CN(C(c3ccc(C(C)O)cc3)=O)C2)ccc(S(N)(=O)=O)o1 c1(OCC(=O)NC2C(CNC(c3cnc(C(C)(C)C)[nH]3)=O)CC2)ccc(Cl)cc1F C#CC1(C(=O)N(C2CCCC2C)C)CCN(C(=O)C(C)C(C)C)C1 CC1CCN(C(=O)CC(C)C(C)(C)C)CCN1C(=O)Cc1cccs1 CC(C)C(C)(CNC(c1cccc(Br)c1)=O)NC(c1ccc(C2CC2)nc1)=O C1(C(N(C2CCN(C(=O)CCCNS(C)(=O)=O)C2)CC)=O)COC(C)C1 C1(C)(CNC(C)CC2CCC(=O)N2)CCN(C(=O)C(CO)c2ccccc2)CC1 N1(C(CCC=C=C)=O)CCCC12CCCN(C(c1cccc3nccn13)=O)C2 c1(C(C)NC2CCN(CCC3CCOC3)C2)ncc(Cl)n1C CN1C(=O)CSC1=CC(=O)NCC(C1CCN(C(C2(CO)CCCO2)=O)CC1)F CCC1=NOC(CC(=O)NCC(c2ccccc2)CNC(c2cnns2)=O)C1 c1(OC)ccc(CCCCC(=O)NCCCCN(C)C(c2csnn2)=O)cc1 C12(NC(=O)CC3CCCOC3)CCCN(C(c3cc(F)c(F)cc3F)=O)CC1C2 c1(C(=O)NCC(c2cccc(C)c2)NC(CCCOC)=O)scc(C)c1C C1(C(=O)NCC(C)CNC(c2cc(C3CC3)[nH]n2)=O)CC12CCC(C)(C)CC2 C(=O)(C1CCCc2sccc21)NC1CC(SCC(=O)NC2CC2)C1 Cc1ccnn1CC(N1CC(CNC(c2ccn(C(C)C)n2)=O)C1)=O C1(NC(CCc2cn(C)nc2)=O)CC(NC(=O)C=Cc2cnc[nH]2)C(O)C1 Cc1nc2cc(C(=O)NCC3CCCCN(C(C4CC4C#N)=O)C3)ccc2s1 c1(CC)ccc(OCC(=O)NC(C)CN(C(=O)C(c2csc(C)n2)C)C)cc1 c1(C(=O)NCC(CC=C)NC(C2(F)CCCOC2)=O)c[nH]c2c(C#N)cccc12 C1(OC(F)F)CCC(C(=O)N(C(=O)COCCN(C)C)C2CC2)CC1 CC1(C)NC(=O)OC12CCN(C(c1nnc(C3CCCC3)s1)=O)C2 CN1N=CC(CC(C(=O)CC(C)c2cnn(C)c2)=O)C1=O.C1(OCCN)CNC1 N1(C(C2(NC(=O)CCc3cscn3)C(C)(C)C2)=O)CC2(C1)CC2(F)F C1(CC(=O)N(CC(C)(C)C)CC)CCC2(CC2)C1.C1(CC(=O)OCC)CCCCO1 CS(=O)(=O)CCC(=O)N1CC2C(CNC(=O)C(O)COCc3ccccc3)C2C1 c1(OC)ccc(CC(=O)NCC(C)N(C(=O)C(c2cccnc2)C)C)cc1F C1(CN(C(CCN(C(C(CSC)OC)=O)C(C)C)=O)C)CCN(C)CC1 N1(C(C(CCC)C)=O)CC2CN(C(c3c(C)ncnc3C)=O)CCC12 c1(OC)nccc(C(=O)NCCC2CCCN2C(C2CCCC(OC)C2)=O)n1 c1(C(C(=O)NCCOCC)N(C(C)CSC)C)ccncc1OC c1(NCC(CC)CC)ccc(S(=O)(=O)NC2CC(O)C2(C)C)c(Cl)c1 N1(C(C(CCC)OC)=O)CC(NC(=O)CC2SC3=NCCN3C2=O)CC2(CC2)C1 C1(N(CCCC)C(C2CC=CC2)=O)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 C(=O)(C(C)C(C)(F)F)N(C)CC1N(C(C(CC=C)NC(C)=O)=O)CCCC1 C#CC1(C(=O)NCCCn2ccnc2)CN(C(=O)Cc2n[nH]c(C)n2)C1 C(C(COC)C(=O)N1CCC(C(C)NC(=O)CC2CCCCN2C)CC1)OC C1(O)(CNC(=O)OC(C)(C)C)CCS(=O)(=O)CC1.C1(C)C(C(C)C)C(=O)N1 C1(C(=O)NCC2CCCN(C)C2)CC(O)CCN1C(=O)CCc1ccc[nH]1 c1(CCC)sc(C(=O)N(CCCNC(=O)C=CS(C)=O)C)cc1CC Cc1ccc(OCC(=O)O)c(NC23CCC(CC2NC(=O)CC2CC2C)C3)c1 c1(CC(N2C(C(=O)OCC)CC2C)=O)ccc(O)cc1Br C(=O)(CCCCN(C)C)NCC(C)(C)OCC(=O)NCC1(O)CC(N(C)C)C1 c1(CNC(C2CCN(C(=O)C(F)(F)F)CC2O)=O)cccc(Cl)c1[N+](=O)[O-] C=CC(C)(O)C(=O)NC1CC(C(=O)NCCc2cncc(C)n2)C1 C(=O)(C(C#N)(CC)NC(C1CC1COCC)=O)c1cn(CC(COCC)O)nn1 C12(CNC(CCOCC#C)=O)CCCC1N(C(=O)CCBr)CCC2 C(C)(CCCCNC(=O)C(C(C)C)c1ccncc1)NC(c1c(C)con1)=O C1(CNC(C(COC)N(C)C)=O)CC2CCC1N2C(=O)C=C(C)Cl C1(C(=O)NCC(C2CC2)NC(COC(CC)C)=O)CCc2cncn2C1 c1(C(N2CCC(CN(C(CC(=O)NCC)=O)C)C2)=O)cnc2c(c1)NCC2 C1(CC)CN(C(=O)CO)CCN1C(=O)C(CCOC)OC.c1(C(=O)NC)ccc(C)s1 N1(C(C2CCN(CC)C2)=O)CCOC(CC(=O)NC(C)(CC)CC)C1 c1(C(CCC(=O)NC2CC(CNC(C3C(C)C3)=O)C2)=O)csc2ccccc12 N1(C(C(C2CC2)OCC)=O)CCCC(C(=O)Nc2ccc(CO)c(Cl)c2)C1CC Cc1cc(Cl)ncc1CC(=O)N(CC(C)NC(C1CCC(OC(F)(F)F)C1)=O)C CC(C)CC(=O)C(=O)NC(c1nocc1C(=O)NCCc1cnco1)C C(=O)(CC(CC)NC(=O)C(CCOC)OC)NC(COC)COC C1(C)(C(=O)NCCCCN(C(CCCNC(=O)NCC#C)=O)C)CCC12CCC2 c1(OCC)cc(C=CC(=O)NC(c2ccc(F)cc2)CC)ccc1N C(=O)(CCS(C)(=O)=O)NCC#CC(=O)NC(C)Cc1ccsn1 CC1CN(C(C2CSCCN2C(=O)CCc2ccn(C)c2)=O)Cc2nncn21 CC(C)CC(O)C(=O)NC1CCC(C)(CNC(=O)Cc2cc(C3CC3)on2)CC1 N1(C(CCSCCCC)=O)CCN(C(=O)C2=CCOCC2)CC12CC2 Cc1ccc(O)c(C(N2CCC23CN(Cc2ccc(O)c(I)c2)C3)=O)c1 c1(OC)cccc(OCC(=O)NCC2CC(NC(=O)C(C3CCC(=O)N3)C)C2)c1 C1(NC(C2(C(N(C)C)=O)CC2)=O)CCC2CCN(C(c3[nH]ccc3C3CC3)=O)C12 N1(C(C=C(CC)CC)=O)CCCC1C(C)(C)NC(c1ccc(COC)s1)=O C(CS(=O)(=O)CC(=O)N(C1CCN(C(c2csc(F)c2)=O)CC1)CCO)OC Cc1nnc2n[nH]c(N3CCCCC3C(N3CCNCC3)=O)c2c1C c1(C(N(CCCN(C(COC(CC)C)=O)C)C)=O)c(F)ccc2ccncc12 C1(NC(C(COC)OC)=O)CC2(CCN(c3nccc(C(C)(C)C)n3)CC2)C1 C1(CC=C)COCC1NC(C1(NC(=O)C(F)(F)C2CC2)CCC1)=O Cc1cc(C2CC2)ccc1C(=O)NC(C)CCCNC(C1CCCOC1)=O CC(C)C(C(=O)NC(C)CCN(C(=O)C(C)(C)CCF)C)C(C)C C1(C(=O)OCC)CN(C(c2cc(OC)cc([N+](=O)[O-])c2)=O)CC12CCOCC2 C1(CC(=O)NC2CC2)OC(C)(C)OC1=O.C12(CC1)C(=O)N(C)C1CC1NC2=O C#CC1(O)CCCN(C(=O)CC2CCN2C(=O)C(=O)NC2CC2)C1 c1(NC(C2CN(C)C(=O)CC2)=O)ccc2c(c1)C(N)CC2 C1(NC(C2CC(n3cc(CC(C(C)C)(C)O)nn3)C2)=O)CCOC2(CCC2)C1 c1(C(=O)NCC(CC)SC)ccc(C(=O)Nc2cccc(C(C)C)c2)cc1OC C1(CNC(Cn2ncc(C)c2)=O)CN(C(=O)CNC(=O)OC(C)(C)C)CCCO1 Cc1c(C(=O)NC2(CO)CCN(C(c3csnn3)=O)C2)cnn1CC(F)F CS(=O)(=O)c1ccc(NC(=O)CC(C(=O)OC)c2cccs2)cc1F Cc1nc(C(=O)NC2CCN(CCNC(C3CCC3C)=O)CC2)c(C)s1 N1(C(CSC(C)C)=O)CC(CO)C2(C1)CN(C(=O)CC1CCCC1)C2 c1(OC)cc(N)c(F)cc1C(N1CCCC(NC(C2CCN(C)C2C)=O)C1)=O O=C(NN1C(=O)NCCC1=O)c1cncn1C1CC1 C(c1ccc(Cl)s1)=CC(=O)NCc1ccc(CNC(c2cc(F)n[nH]2)=O)cc1 C1(CCC(=O)NCC(C)(C)NC(CCN(CCCCC)C)=O)CCC(=O)C1 C=CCC(C)(CC=C)NC(=O)CCN(C(=O)C(CCC)N(C)C(C)=O)CC C1(C(=O)NC2C3CN(C(C(C)NC(N)=O)=O)CC2C3)CC2CC(O)CC(C1)C2 c1(C(=O)NCC23CC(c4ccccc4)(C2)C3)c[nH]c2ccc(Br)cc12 C1(C(=O)NCC2CC(NC(C(C)c3ccsn3)=O)C2)CCOC2(CCCCC2)C1 C1(NC(C(C)N(CC)CC)=O)CC2CC(C1)CN(C(=O)CCC1CCCCO1)C2 N1(C(C(CSC)OC)=O)CC(NC(c2c(C)noc2C(F)(F)F)=O)C(SC)C1 N1(C(C(C)NCCCCCC)=O)CCOCC1C CC(C)CS(=O)(=O)CC(=O)NC1CCN(CCCNC(C2CCCC(F)C2)=O)C1 c1(OC)cc(-n2nc(C3CCCC3)nc2C(C)SC)cc(F)c1F C1(C(=O)NCC(C)O)CCOCCN1C(=O)CC(C)(C)O N1(C(c2ccc(C(=O)NC3CC4(CCC4)CO3)cc2)C2CC2)Cc2ccccc2C1 CCCCCCCCS(=O)(=O)N1CC(N(C(=O)COc2ccccc2C)C)C1 CC1OCCOC1C(=O)NCC1(CO)CCN(C(C2C=CCC2)=O)C1 c1(C(N(CC(C)(C)CNC(=O)C(F)C2CC2)C)=O)c(Br)cncc1[N+](=O)[O-] CCC(C)CCC(=O)NC(C)(C)CN(C)C(c1cccc(COC)c1)=O C(=O)(CCCCN(C)C(C1CCCC1)=O)N(C(C=C)C1CC1)C C12(C(=O)NCc3n(CCC)ccn3)CC(CN(C(=O)CCCC(OC)OC)C1)C2 N1(C(c2ccn(CC)n2)=O)CCOCC1CC(=O)NCC(C)(O)C1CC1 C1(C(N2CC(CCOC)C2)=O)CCC(NC(=O)CSc2nc[nH]n2)CC1 CC(CCC(C)(C)C)C(=O)N1CC2CCCC2C1C(=O)NCCc1ccccn1 C1(C(N)=O)(CNC(C2(C(C)(C)O)CC2)=O)CN(C(=O)COCP(C)(C)=O)C1 C(=O)(CCCCCF)NCC1(C(C)NC(c2ccc(OC(C)C)nc2)=O)CC1 c1(CC)ccc(C(=O)N(C)C)c(C)n1.c12cn(nn1)CC(=O)N(CC)C1CC2C1 N1(C(C(COC(C)=O)C)=O)Cc2nccn2CC(NC(=O)CC2(C)CCCO2)C1 N1(C(C(CSC)OC)=O)C2CCCC1CN(C(c1cc(C#N)c[nH]1)=O)C2 C(C(CC(C)C)NC(C1CCCN1CC)=O)NC(C=CCC)=O N1(C(CC(C)(C)C)=O)CC2(CNC(c3ccc(Cl)cc3)=O)CC1CO2 C(C(C)(C)C(=O)NCC(C(C)(C)C)NC(=O)C(C)CN1CCOCC1)NC(C)=O c1(C(N(CCN(C(c2c(CC)nn(C)c2Cl)=O)C)C)=O)ccc2sccc2c1 C1(C)(CNC(C2C(OC)CCC2)=O)CCN(C(=O)Cc2nocc2C)C1 c1(C(=O)NC2C(NC(c3cccnc3O)=O)CCCC2)cc2c(nn1)OCCS2 c1(C(N2CCC(C)(C#N)CC2)=O)cc2c(s1)CCN(C(C1CCC(O)CC1)=O)C2 N1(C(c2n(CC)ccn2)=O)CCN(C(=O)Cc2cncs2)CC2CCCCC12 C(=O)(CC1OCc2ccccc21)NCC(CNC(=O)CCSc1ccccc1)O N1(C(c2cnc(C)s2)=O)CCC(NC(C2(F)CCS(=O)(=O)C2)=O)CC1C c1(CNC(C2N(Cc3cccc(C#C)c3)C3C(C2)C3)=O)cccc2[nH]ncc12 c1(C(=O)OC)cccn(CC(=O)NCC(C(C)(C)C)NC(=O)C=C2CC2)c1=O c1(C(=O)NC(C)CN(C)C(c2ccn3c2CSCC3)=O)cc2nn[nH]c2cc1F CCCC(C(=O)N1C(C(=O)NC(C)(C)C(=O)OC)CC2CC12)OCC Cn1[nH]c(=NC(=O)C2CC(F)CN(Cc3cc(Cl)cnc3Cl)C2)cc1Cl CCCC(CNC(=O)CC1CCC(=O)N1)C(=O)N1CCCC1(C(C)C)CO c12cnc(F)cc1C(=O)N2C.c1(NC(=O)OCC)c(C)cccc1Br C(=O)(C1CCc2ccccc21)N1CC(NC(CCc2c(C)noc2Cl)=O)(CF)C1 C1(CNC(CC(CC)(F)F)=O)CN(C(c2occc2CC)=O)CC12CCC2.C(C)C c1(C(N2CC(NC(CCC(C)SC)=O)C(C(F)F)C2)=O)cc2ccc(F)cc2o1 N1(C(C(C(C)C)=O)=O)CC(C(N2CC(O)CC2(C)C)=O)CC(F)(F)C1 Cc1cn2cccc(C(=O)NCC3CN(C(=O)CCC(C)N(C)C)CCO3)c2n1 N1(C(c2c(CC)n(C)nc2)=O)CCN(C(=O)C=Cc2ccn(C)c2)C2CC12 c1(C(=O)NC2C(CNC(C3C(=C)C3)=O)CCCC2)[nH]c2ccccc2c1C#N Cc1ccc(N)c(C(=O)NCC23CC(NC(=O)CCC4CCC4)(C2)C(C)O3)c1F c1(C(N2CCC(OC)(CNC(=O)C=C3CCOCC3)C2)=O)cnc2ncccn12 CN1CCN(C(c2ccsc2NS(C)(=O)=O)=O)CC1CNC(C12CC(O)C1C2)=O C(C(CC(=O)NC1(CO)CC=CC1)NC(c1nonc1N)=O)OC C1(NC(CC2CN(C)CC2O)=O)CCCCCN(C(=O)Cc2cncc(F)c2)C1 CCCC(O)C(=O)NC1(CCO)CN(C(c2ccnnc2NC2CC2)=O)C1 c1(C(=O)NCC2CCCN2)ccc(F)c(S(N)(=O)=O)c1 N1(C(c2cnc(OC)s2)=O)CCOC(CNC(=O)CC2CC3CCC2C3)C1 CC(CC(C)(C)C)C(=O)N(CCCN(C)C(c1ncn2c1COCC2)=O)C C1(S(N)(=O)=O)(C(=O)NC(CCNC(c2cc(C)oc2C)=O)C)CCCC1 c1(C(=O)OCC(=O)NCC(CNC(COC)=O)F)cc(C(C)OC(C)(C)C)no1 c1(OC)cccc(CC(=O)NCC2(F)CC(NC(=O)C=C(C)C)C2)c1Cl C1(NC(=O)Cn2cnc(Br)n2)CCN(C(=O)CCn2cncn2)CC1O c1(C(=O)NC2C(C)CCN(C(=O)C(C)(F)F)C2)cc2n(n1)CCNC2=O c1(CC(N2CC(C)C(NC(C3CC3C(F)F)=O)C2)=O)cccc(C#N)c1 c1(C(C(=O)NCC=C)N(CC(F)F)C(C)C)cc(Br)no1 N1(C(C(C)O)=O)CC(C2CCCCN(C(c3cc(C4CC4)sn3)=O)C2)C1 N1(C(c2onc(CC)n2)C)CCC(NC(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C(C)(C)C1 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)NC(C1CCCC1)C#N N1(CCNC(C(c2cnn(C)c2)NC(c2c(C)non2)=O)=O)CCOCC1=O C=CCCC(C)(c1nnnn1CC(F)F)NCC1(c2ccccc2Cl)CCC1 Cc1nc(NC(C2C=CCN2Cc2ccc(F)c(I)c2)=O)ncc1Br c1(N(C)C)ccc(N)c(C(=O)NC2CC(NC(c3c(Cl)cncc3Cl)=O)C2)c1 C12CCC(O1)C(=O)N(CCNC(C)=O)CCNC(=O)C2.O(C(F)F)CC c1(NCCC2N(C(c3cnccn3)=O)CCCC2)nc(Cl)nc2[nH]c(O)nc12 c1(C(N(C(C)C)CCNC(c2sccc2C(F)F)=O)=O)cccc2c1COCC2 CC(CC(=O)N1CCOC2(CCC2)C1)C(C)(C)NC(=O)CC1CNC(=O)O1 C1(NC(C2(CC)CC2)=O)CN(C(C2CCC2(C)C)=O)C2CCCCC12 Cc1cc(C)n2nc(C(=O)N(CC(C)NC(c3ncncc3C#N)=O)C)cc2n1 N(C)(C1CN(C(c2cc(C)n(C)c2)=O)CCc2ccccc21)C(CC=CC=C)=O C1(CC)CN(C(=O)C(=O)NCC2CC3CCC(C2)C3)c2ccccc2O1 c1(C(N2CCCC(CC)(NC(=O)Cc3cncs3)C2)=O)cnc2ccccc2n1 C1(CC(=O)NOC2CCOC2)CCCC12CC2.c12cn(nn1)C2 CC(Cc1cn[nH]c1)CN=c1nc(N2CCC(C)C2)c2cc(N(C)C)ccc2[nH]1 N1(C(C(C(C)O)C)=O)CC2CN(C(c3csc(=N)[nH]3)=O)CC(C1)O2 N1(C(C(C(=O)OC)OC)=O)CC2CN(C(C34CCC3CC4)=O)CC2C1 Cn1cc([N+](=O)[O-])cc1C(N1CCCC1C1(O)CN(C(C2C=CCCC2)=O)C1)=O N12CCC(C(C)(C)C1)C(=O)NOC(CC(C)C)C2=O.C(CCC(C)C)=CC Cc1ccc(CNC(C23CC2CN(S(=O)(=O)CC#N)C3)=O)c(I)c1 CCCCC(CNC(c1coc(C(N)=O)c1)=O)NC(=O)Cc1cnc(C)s1 c1(C(=O)NCC(C)N(C(CCCN(C(C)=O)C)=O)C)cc(C)cc(O)c1 C1(CNC(C(C2CC2)OC)=O)CCN(C(=O)CCOCC2CCC2)C1 Cc1cncc(C(N2CCOC(CCNC(=O)Cc3ccc(C)s3)C2)=O)n1 c1(NC(C2(CC)CCC2)=O)cncc(-n2cccc2)n1 c1(C(N(C)CC2CCN(C(c3cccc(F)c3)=O)C2)=O)nccn2cnnc12 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(C2(CO)CCC2)=O)CCC(C)(C)C1 c1(C(N2C3C(NC(c4nc(C)nc(O)c4)=O)CC(C3)C2)=O)c(F)ccc(Br)c1F CC(C)(F)CN=C1NC(=O)N2CCCC3(CCN1OCCC3)CC2.C1(C)CC1 N1(C(c2cc(C)sn2)=O)C2CCC1CC(C(N1CCC3(CCCO3)C1)=O)C2 C1(CC(=O)NCCC2CC(C(=O)NC3CC3c3cncs3)C2)CCCOCC1 N1(C(C=C2CCN(C)C2)=O)CC(O)CC1CNC(=O)C(C)(C)c1ccnn1C C#CCC(C)(C(=O)N1CCC(O)C(CO)C1)NC(=O)CC1COCCOC1 C=CC1(CC(=O)NCC(C)OC(F)F)CN(C(c2coc(C(F)F)c2)=O)C1 c1(-n2cc(CCCC(=O)NC(CC(CC)C)C(=O)O)nn2)c(F)c(F)cc(F)c1F c1(C(N2CCCCC2CO)=O)cc(Br)c(F)cc1Cl.N12CCC1C2 c1(C(=O)NC2CCCN(Cn3ncc(C#C)c3)C2)ccc2c(Cl)ccnc2c1 N1(Cc2cc(C)nc(C)c2)CC2CC(NC(c3ccc(CO)cc3)=O)CC2C1 c1(N(C(C2(O)CCNCC2)C)C(c2cnoc2)=O)ncc2ccsc2n1 C(CC(C(=O)NC(c1nc(C)oc1C)C)NC(=O)C(C)OCCCOC)=CC c1(CC(=O)NC(C)C(C)NC(=O)CCF)cnn(-c2ccccc2)c1 c1(CN2CC3(C(C(N4CC(=O)NC4)=O)C3)C2)cc(Cl)cnc1Cl n1(CC)nc(C)cc1C(N1CCOCC1CN(C(=O)CCOC1COC1)C)=O C1(C(=O)NCc2ccc(C(=O)OC)[nH]2)CC12CCN(Cc1ccc(Cl)cc1Br)C2 C(c1cnc(C)nc1O)=CC(=O)NC1CC(CNC(c2oc(CC)c(C)c2)=O)C1 c1(C(N2CC(CC(=O)NCC#C)C3(C2)CC3)=O)ccnc2ccccc12 c1(C(=O)NC2CCN(C(CCCC(=O)OCC)=O)CC2F)nsc2ccccc12 CCC(C)(COC)CN=c1[nH]c(=NCc2nc(C(N)=O)cs2)c2ccccc2[nH]1 N1(C(c2c(C)csc2C)=O)CCN(C(=O)NC2CCC3CC23)CC1C#N c1(C(N2CCC(NC(c3cc(OC)ncc3)=O)C2)=O)ccc(C#N)nc1O c1(CC(=O)N(C2CCC(NC(c3ccnnc3)=O)C2)C)ccc2nn[nH]c2c1 CC1CN(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CCC1N(C(=O)Cc1nc[nH]n1)C C(CN=c1[nH]c2c(c(=NCC3(CO)CC34CCOCC4)[nH]1)CCC2)N(CC)CC Cc1ncc(C(=O)NCCc2cn(CC3CCC4CC4C3)nn2)c(O)n1 Cc1cc(NCC2CCCN(C(c3cocn3)=O)CC2)n2ncnc2n1 C12CC3(C1)C(C31CCC1)C(=O)N2.C(=O)(C1CCCN(C(=O)OC)CC1)NC(C)(C)C CCCC(O)C(=O)NCC(CC)NC(=O)CC1(C(F)F)CC1 N1(C(C(C)=C2CC2)=O)CC(CNC(c2ocnc2-c2ccccc2)=O)CCC1C c1(C(N(CCOCC(=O)OC)NCC)=O)ccc(Cl)cc1 N1(C(C2(OC)CC(C)C2)=O)CCC(NC(C2CC23CCOCC3)=O)C2(CCC2)C1 CC1(C)CCC(C(=O)NC2CC(NC(c3ccc(O)c(F)c3)=O)C2)CC1 N1(C(c2cc(CN(CC(C)C)CCCC)[nH]n2)=O)CC(O)CC1C(=O)NNC=O.CC CC1(C)CCC(C(=O)NC2CC(C)(C)OC2=O)(NC(=O)COC2CC=CC2)C1 N1(CC(=O)NC(C(CSC)c2ccccc2)=O)CCC(C)=C(Br)C1 c1(C(=O)NCC(CC)NC(=O)CN2CCCCCC2)cnc2n1CCCCC2 CC(C)C(C#N)C(=O)N1CCC(CCC(N2CCCN(C(C)C)CC2)=O)C1 Cc1cc(Br)c2ncnc(OCCCc3cccs3)c2c1 c1(C(=O)NC2(C)CN(C(C(CC)Sc3ccccc3)=O)C2)nc(C(C)C)sc1C C1(COC)CC(CNC(=O)C(c2ccc(Cl)cc2)=O)N(C(=O)Cc2cnns2)C1 c1(OCC)ccc(C(=O)NC2CCCN(C(C3CC3C)=O)C2)cc1C(F)(F)F CC1CCN(C(=O)CCOC2CCC2)C(CNC(C2CC3CC(=O)C2O3)=O)C1 Cc1nc(Cl)c(NCCC2CN(c3ccc([N+](=O)[O-])cn3)CCS2(=O)=O)c(Cl)n1 N1(C(C2CC(N(C)C)C2)=O)CCC(C(N2CCC3(CCCO3)C2)=O)CC1(C)C c1(C(=O)NCC2(NC(C(C)Cn3cccn3)=O)CC2)cc2n(c1)CCOC2 c1(N(C(CCOC)=O)Cc2ccc3c(c2)OCCO3)ncnc2cccnc12 c1(OC)nsc(OC)c1C(=O)NCC(C(C)C)NC(=O)C(n1cc(C)cn1)C N1(C(CCOCC)=O)CCC2CCN(C(=O)C(c3ccccc3F)(C)C)CC2C1 C1(C(N2CCN(C(c3cc(C)no3)=O)CC2)=O)Cc2ccccc2C1C C1(C(=O)NCCc2c(C)nc[nH]2)CN(C(C2CCC(C3CC3)C2)=O)CC(C)O1 c1(C(=O)NC(CC)(CC)C(F)F)c(Cl)cc(I)c(F)c1F C(=O)(C(=O)C(F)(F)F)OC(=N)O.C12CCC(CC1)C(C)n1cc(nn1)CC2 C1(NC(c2nc(OC)c(C)s2)=O)CCN(C(c2cc(C(F)F)n(C)n2)=O)C(C)C1 c1(C(=O)NCC(=O)NC2C(SC)CCC2)c(Cl)cnn1C.C12(CCC1)C(=O)NC2 CC1CN(C(=O)CCN(C(c2ncccc2O)=O)C2CC2)CC(=O)N1 CCCCC(CC(=O)NCC1CCCSC1(C)C)N(C(=O)OC(C)(C)C)C1CC1 CC1CN(C(=O)CC(C(F)(F)F)c2ccccc2C(=O)O)CCC12CCOCC2 C(=O)(CC1CCc2ccccc21)N1C(C)(C)CC(NC(=O)CCCC2CCC2)C1 C#Cc1cnn(CC(=O)NC(CNC(=O)COCCc2cccs2)(CC)CC)c1 C1(C(=O)NCCC(O)CNC(=O)C=CC(C)(C)SC)(OC)CCC(C)(C)CC1 N1(C(CN(C)C2CC2)=O)CCC(C)(C)C(NC(c2cc(C(N)=O)ccc2F)=O)C1 C1(C)(C(=O)NC(C)(C)C)CCCN(Cc2ccnc(-c3ccc(CO)cc3)c2)C1 c1(N2CCC(OC)C(C)(C)C2)nc(=NCc2cn(C)nn2)[nH]c2ncn(CC)c12 C1(NC(Cn2c(C)cnc2)=O)CCCCN(Cc2nc(C(C)C)no2)C1 C(CC)(CCCC(=O)NCC[Si](C)(C)C)NC(C1(CC=C)CCC1)=O CCC(C)CC(=O)N1CCC(CCC(=O)NCC2(C)CCCO2)CC1 C12(C(N3CC4C(CNC(CCC(=O)NCCC)=O)C4C3)=O)CCCN(CC1)C2 N1(C(c2ccc(N(C)C)cc2)=O)CCn2c(CNC(C3(O)CCC3)=O)nnc2C1 N1(C(CCOCCOC)=O)CCC(O)(C(C)NC(c2cc(C(C)=O)cn2C)=O)C1 c1(C(=O)NCC23OCC(NC(C(C=C)O)=O)(C2)C3)cc(F)cnc1O C1(C(=O)NC2(CNC(c3cccc(C)c3)=O)CCCC2)CN2CCN1C(C)C2 N1(C(CC(C(C)C)NC(c2ccc(CC)s2)=O)=O)CCC2(CCC2)C(O)C1 c1(SCC(N2CC3C(NC(C=CC(=O)OCC)=O)(C3)C2)=O)ccc(C)cc1C Cn1cc2ccc(C(=O)NC3COCCN(C(=O)C(C)(C)CCl)C3)cc2n1 CC1CC(NC(c2ncoc2C2CCC2)=O)CN(C(=O)C=C2CCN(C)C2)C1 N1(C(C(C(C)O)N(C)C)=O)CC2(C1)SCCC2NC(c1cc2cnccc2o1)=O N1(C(C(CC)C#N)=O)CC(C2CCCN(C(=O)Cc3ccco3)C2)C1 N1(C(CSCC(C)C)=O)CCC(CF)(NC(=O)C(C)Cc2ccccc2F)C1 CCCCC(C(=O)N(C)CC1CCCN1C(c1ccc(O)c(Cl)n1)=O)NC(N)=O C1(C)(COC(Cc2c(-c3ccccc3)nc(C)s2)=O)Oc2ccccc2O1 c1(CN2CCC(O)(C(=O)Nc3ncc(C)nc3Cl)C2)ccc(I)c(F)c1F c1(C(N(CCOCCN(C(=O)CN(C)S(N)(=O)=O)C)C)=O)nccc2n[nH]cc12 Cc1sc(C)c2sc(C(=O)NC3CN(C(=O)CCCC(N)=O)CC4(CC4)C3)cc12 N1(c2ncnc(NC3C(CC=CC)COC3)c2C)CCC2(CC1)CCN(C)C2 C1(C)(CCNC(CCC=CC)=O)CCN(C(=O)C(C)Cc2ccc(O)cc2)C1 C1(C(N(CC(C(=O)NC(C)Cc2cn(C)cn2)C)C)=O)CCNC(=O)C1 C(=O)(C1=COCC1)NCCCN(C(c1ccc(C2C(C)C2)o1)=O)CCO N1(C(C2C(OCC)C2)=O)CC2C(N(C(=O)CCc3ccsc3Cl)C)C2C1 N1(C(c2nc(CC)oc2C)=O)CCCC1C1CCCN1C(c1cccnc1C)=O N1(CCN(CC(N2CC(C(F)(F)F)C2)=O)C)CC2CC(O)CC1C2 c1(OC)cc(C(N2CC(O)(C3CCCN3)C2)=O)sn1 C#CC(CC(C)(C)C)NC(C1CCCN1C(=O)C(C)OCCCC)=O Cc1cc(CNC(=O)CCCN(C(=O)CC2CCC(=O)N2C)C)oc1C N1(C(C(=O)OC)=O)CCN(N2CCC(C(F)(F)F)C(OC(C)C)C2)CC1 Cc1nc(O)sc1C(=O)NC1CCCCC1CNC(c1ccc(C(F)F)o1)=O C(=O)(C(=O)N=S(C)(C)=O)NCCN(C(c1ccc(CN(CC)CC)o1)=O)C1CC1 CCC(C)(CCC(C)C)C(=O)N1CCn2nc(CNC(C3CCOC3)=O)cc2C1 C(=O)(C(O)C1=CCCCC1)NC(C)(CO)C(=O)NCC1(O)CCOC1 S(=O)(=O)(c1cccc(C#N)c1F)Nc1sc2ccc(C)cc2n1 c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC(F)C2)=O)cc2cccn2cn1 Cc1ccc2c(=NC(C)c3cc[nH]n3)[nH]c(=NCCCC3CCOC3)[nH]c2c1 S(=O)(=O)(c1cccnc1N)NC.Cc1ccccc1C(O)CCCCCCCF CC12CCC(C(=O)NCC3CC3NC(c3csc(-c4ccoc4)n3)=O)(C1)OC2 CC(C)(CCCNC(c1cc(F)c[nH]1)=O)C(=O)N1CC(S(C)(=N)=O)C1 N1(C(C(CSC)C)=O)CCC(N(C)C(c2coc(C3CCCCC3)n2)=O)CC1 C(C)(C(=O)NC1CC(OCC(=O)NCCc2cccs2)C1)OCOC C1(C(=O)NC(C)CCO)CCCCN1C(C1(OC(=O)C2CC2)CC1)=O c1(OC)ccc(CN2CCCC2)cc1-c1cc(F)ccc1C.N12CCC(C1)C2 C1(NC(C2CC23CCC3)=O)CCN(C(=O)CC2CCOCC2)C(C2CC2)C1 c1(Cc2n(CCCOC)nc(-c3cccc(OC)n3)n2)noc2c1CCCC2 c1(OC)ncccc1C(N(CC(CNC(c1cnn(C2CCC2)n1)=O)C)C)=O c1(C(N(C(C)CNC(C2CCC(C)O2)=O)C)=O)ccc2ccnc(O)c2n1 C1(NC(C2(CCC=C)CC2)=O)CN(C(=O)C=C(C)CCC)CC1(C)C CC1C(NC(=O)CC2OCCOC2(C)C)CCCN1C(c1nn(C)cc1Cl)=O CCCCN=C(NCc1ncccn1)NNC.C1(C)CCC2(CC1)CC2 C(C(C)(C)C(=O)NC(C)CC(C)O)NC(CC1(NC(C)=O)CC1)=O N1(C(C(=O)NCC2CC2)=O)CCOC2CCN(C(C3CCCNS3(=O)=O)=O)CC12 c1(C(N(C)CC2CCCN(C(=O)Cc3c[nH]nc3O)C2)=O)cc(O)ncc1Br C(=O)(C1COc2ccccc21)NCC(CC)(CC)NC(=O)C(O)CC1CC1 C1(NC(C(C)C2CCCO2)=O)CN(C(=O)C(=C2CCCCC2)F)C2CCCCC12 N(C(=NCCCF)N1CCSC(C(F)(F)F)C1)CC(=C)CCC1CCCCC1 c1(C(N(CCCNC(C(c2ccnn2C)C)=O)C)=O)[nH]cc2c1CCCC2 N1(C(C2C(C(C)O)C2)=O)CCC(NC(c2cncc(Cl)c2Cl)=O)C2(CCC2)C1 c1(C(=O)NCC(C(C)C)NC(C2C(C=C)C2)=O)cnc(C)nc1C CCCC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)Cn2cc[n+](C)c2)C1 c1(C(=O)NCC2(O)CC(CNC(C3C(C)(C)C3(F)F)=O)C2)ccc(O)nc1Cl N1(C(CCC2(C)CC2)=O)CCC(c2nnc(CNC(=O)CC(C)(F)F)s2)CC1 N1(C(C=Cc2cc(C)no2)=O)CCC2CCC(C1)N2C(=O)Cn1cncn1 c1(C(N(C2CCN(C(c3cccnn3)=O)C2)C)=O)ccc(C(C)(F)F)nc1O c1(C(N2C(CN(C)C(C3(F)CCOC3)=O)CCC2)=O)ccc2c(c1)COCC2 C(C)(C(=O)N1CC(CCNC(c2ccnc(F)c2O)=O)C1)(C(C)C)OC c1(C(=O)NCCC2CCN(C(C=CCCC)=O)C2)ccc2ccc(Br)cc2c1 C1(NC(CCc2ccc(C(=O)NC(CCC)CCO)[nH]2)=O)CCC(F)(F)CC1 CC(CC(=O)NC1CC(C)N(C(=O)COc2ccn(C)n2)C1)CC(F)(F)F CCCCCCC(C)NC(C1(NC(=O)C=C(C)c2ccco2)CCCC1C)=O c1cc(N(C(COCCOCC#C)=O)CC)no1.C1(CO)CC(CCN)C1.CC.OC Cc1cc(C(=O)NC23CCC(NC(C45CC(CO4)C5)=O)(CC2)C3)ccc1F C#CC1(C)COCCN1C(c1ccc(-c2ccccc2)s1)C(=O)NC CCCC(C(=O)NC1CN(C(=O)Cc2nocc2C)CCC1C)C(C)C c1(C(N(CC(CCC=C)O)C)=O)cc(C#N)cc(C#N)c1 c1(C(=O)NCC2(C(=O)Nc3c(C(=O)OC)cncc3)CC2)cccc(OC)c1F C(CCN=c1nc2scnc2c(N2CCC(CO)C2)[nH]1)N(C1CCC(C)CC1)CC Cc1cncc(CNC(C2CC(O)CN2C(=O)C=C2CCOCC2)=O)c1 N1(C(C23CC(C)(C2)C3)=O)CCCC2C1CCN2C(C1CCC2(CC1)CC(O)C2)=O c1(CC2N(C(C(C)N(CCC)C3CC3)=O)CCC2)cccc2ccccc12 C12(CNC(C)=O)CN(C(c3ccc4c(c3)OCC4)=O)CC(F)(C1)C2 C1(Cc2cn(C(N(C(=O)CCCCc3cnn[nH]3)C)=O)nn2)CCCC(C)(C)C1 N#Cc1cccc(NC(=O)CC2CCN(C(c3cc(O)ccc3I)=O)C2)c1 C1(C(N(C2CCCC2)CCCNC(CCCOCC)=O)=O)Cc2cccnc2C1 N1(C(CNC(=O)NC)=O)CCC(CCNC(c2cccn2C2CC2)=O)C1 c1(NC(C2(C)CCN(C(c3c(Cl)cccc3Cl)=O)C2)=O)c(O)ncnc1O O=C1CC(C(=O)NCC2(CNC(C3CN(C(C)C)C3)=O)CCCC2)C2(CCC2)C1 CCC(CC)C(=O)NOCC(N1CC(C(=O)N(C)C)C1)=O c1(C(N2C(C3(NC(C(CC)NC(N)=O)=O)CC3)CCC2)=O)c(Cl)nn(C)c1Cl Cc1ccc(CNC(C2C3COCC23)c2nnnn2Cc2cccs2)nn1 c1(N2CCCC(C)(CC)CC2)cc(Br)ccc1S(=O)(=O)NCC1CCC(F)(F)C1 c1(NC(C2C(CNC(=O)OC(C)(C)C)C23CC3(C)C)=O)cn2ccc(F)cc2n1 C1(C(=O)OC)C(F)(F)C12CC(C(=O)NCC1CCC3COCC3O1)C2 N1(C(C2CC(O)C(F)C2)=O)CC2CCC(C1)N2C(C1CC(n2ccnn2)C1)=O C1(C(N(CCC(=O)OCC)C)=O)CCN(C(=O)NC)C12CCSCC2 c1(CC(N2CCCC(NC(CC3C(C)=NOC3=O)=O)C2)=O)c(O)nc(=N)[nH]c1C N1(C(C2N(CCC)CCC2)=O)CCOC(CC(N2CCC(F)CC2)=O)C1 c1(OC)cc(CN2CC(O)(CNC(c3cncc(Cl)c3C)=O)C2)cc(Br)c1O C1(C(=O)NC2CCN(c3snc(CCOC)n3)CC2O)Cc2ccccc2CO1 CCC(CNC(=O)COCC(C)(C)C)(CC)C(=O)N(CC(C)(O)C1CC1)C C1(C(N2CC(C(C)NC(C3CCCOCC3)=O)C2)=O)CCCCC1(F)F c1(NC(C(=O)Nc2cccc(-c3ccsc3)c2)=O)cc(Cl)c(Cl)cc1Cl C1(CC)CN(C(=O)CN(c2ccncc2)C)CCN1C(=O)C(C(C)C)OC C1(C(=O)NCCCNC(C(CC)F)=O)CCc2ccccc2O1 c1(NCCNC(=O)NC)nc2ccccc2nc1NC(C1COC(=O)N1)C C1(C(=O)NCCNC(=O)Nc2cccc(-c3ncn(C)n3)c2)(OC)CCOCC1 c1(C(N(C2CCC(NC(=O)C(C)(C)C)C2)C)=O)ccc(P(C)(C)=O)s1 C1(N2C(=O)C3(CC(=C)C3)CCC2)CC(C)OC(C)C1.c1(C(=O)OC)ccn(COC)n1 Cc1ccc(Cl)c(OCC(=O)NC2CC(NC(=O)CC3CCC3C3CC3)C2)c1 c1(C(N(CCCCC(N2C(CCC)COCC2)=O)C)=O)cn2c(n1)CCC2 N1(C(C(C)CO)=O)CC23CCCCC2(C1)CN(C(c1cscn1)=O)C3 c1(OC)cc(N)ccc1C(=O)NC1CCCC1NC(=O)CC1CCC(C)C1 c1(OC)cc(C(=O)NC23CC(NC(=O)C(C4CCCC4)OC)(C2)C3)ccc1C N#Cc1ccc(-c2ccc(NCc3ccc(N4CCC4)cc3)nc2)cc1F c1(CCC(=O)N(CC(C)NC(C2C3CCC23)=O)CC)ccccc1F N1(C(CCC2C(C)(C)C2)=O)CCC2(C1)CN(C(=O)Cc1ccoc1)C2 N1(C(c2cc(OC)cc(F)c2)C(=O)Nc2ccccc2)CCOCC1P(C)(C)=O C1(CCC(N)=O)CCN(CCc2nnnn2CCSc2ccccn2)CC1 CN1CC2CC1CN(C(C13CCN(C(c4ccc(Cl)s4)=O)CCC1C3)=O)C2 c1(C(=O)NCC2(F)CC(NC(C3CC(CC4CC4)C3)=O)C2)cncc2[nH]ccc12 c1(C(=O)NC(CC(C)NC(c2cn(CC)nc2C2CC2)=O)C)cc2ccsc2[nH]1 C(CCCCCNC(=O)C(F)CC)N(C(c1nc(CCC)oc1)=O)C N1(C(Cn2ncc(CC)c2)=O)CC2CCCC2C1C(=O)NCC1CC12CC2(F)F CC1Cn2nccc2CN1C(c1ccc2ccoc2c1)C(=O)NC1COC1 C1(CNC(C2N(C(C(C)NC=O)=O)CCCC2)=O)CC(C)(C)CCO1 c1(C(=O)NC2CCC(C(=O)NCC(F)CO)C2)ccc(I)cc1[N+](=O)[O-] C(CC(C)C)(C(=O)NCCCC(F)F)N(C(C(C(C)C)NC(C)=O)=O)C.C(C)=O Cc1cnc2ccccc2c1C(=O)NCC1(O)CC(NC(=O)COC(F)F)C1 C1(C(N(CCCOC(C)C)C)=O)CC(C)(C)CN1C(=O)CC1COCCO1 CC1CN(C(=O)C(CC(N)=O)NC(C2CCCC(CF)C2)=O)CC(=O)N1C c1(OCC)cccc(Sc2nnc(CSC)n2C)c1 C1(NC(c2c(C)occ2)=O)(CO)CCCN(C(=O)C(C)(C)C)C1.C1C(=O)N1 c1(C(N(C)C)=O)ncccc1C(=O)NCC(C)(C)Nc1sc(N(C)C)nc1Cl c1(-n2c(C3CC3)nc(C(C3CC3)SC)n2)cccc([N+](=O)[O-])c1.c1(C)ccncc1 n1(CC(N2CCCC(C)(CNC(C(CCC)O)=O)C2)=O)c(C)nc2ccccc12 c1(CC)cnccc1C(=O)N(CC(C)(C)CNC(=O)C(C)C1CCCO1)C N1(C(CC(=O)OC)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)C(C2CCC2)C1 C1(F)(C(=O)OCC)CN(C(C2CC23CCC3)=O)C1.C1(=O)C(C2(O)CCC2)O1 c1(-c2nc(C(C)OC(=O)COC3(C)CCCC3(F)F)on2)cccc(C#N)c1 Cc1nc(C)n(CC(=O)NCC2(C)CC(NC(=O)CC3(C(F)F)CC3)C2)n1 CC(C)C(C(=O)NCCc1cncs1)C(C)NC(c1ccsn1)=O c1(CN(C(C)Cc2ccccc2Cl)CC)ncnc2c1nc(CN)n2C N1(C(CCCOCC=C)=O)CCC2(CCC2)C(NC(=O)CC2CCC(=O)C2)C1 C1(CNC(C(C)SC)=O)CCCC2CN(C(=O)C=CC3(C)COC3)CC12 C=C(Cl)CCC(=O)NCC(C12CC(C1)C2)NC(=O)Cc1cccc(C(N)=O)c1 c1(NCC#N)cc[nH]c(=NCCCNC(c2cnn(C3CC3(F)F)c2)=O)n1 C1(NC(=O)NC2CCC3CC3C2)CCCN(c2ccc(-n3ccnc3)cn2)C1 C1(O)(C(=O)NCC2(C)N(C(CC(C)F)=O)CCC2)CCCCCC1 C(C(=O)NC(COC)CC(=O)N1CCCCC1)(C(C)C)OCC N1(C(C2C(C3C(C)C3)C2)=O)CCCC1(C)CNC(c1cc(Br)ccn1)=O C1(NC(COC)=O)CC2(CCN(C(c3ccnc(N(C)C)c3)=O)CC2)C1 C(=O)(C1=CC2(CCOC2)C1)N1CCCC(CCNC(CCCC#N)=O)C1 c1(OC)ccc(Br)c(CN=c2[nH]cc(-c3cc(OC)cc(OC)c3)s2)c1F C(=O)(CC(C)(C)CNC(C1CC(C)(C)C1)=O)NCC(CC)O C1(NC(CN2CCN(C)CC2)=O)CN(C(c2ccc(O)nc2)=O)CC1N=[N+]=[N-] CCC(CCC(=O)NCC(CC)(CC)OC)NC(=O)C(C)(O)COC C1(O)(C(N(C)CC2(CNC(c3cc(C)oc3C)=O)CC2)=O)CCCC(C)(C)CC1 C1(C(=O)NCC2(F)CN(C(c3n(CC#C)ccc3)=O)C2)CCCCC1(F)F N1(C(CC2C(=O)NCC2)=O)CCCCC(CCC(=O)NCC2(C3CC3)CC2)C1 C12(C(=O)NC3CC(NC(c4c(NC)nccc4)=O)CC3O)CCCN(CCC1)C2 Cc1cccc(C(CNC(c2ccc(Cl)cc2)=O)NC(C2(C)CC2C)=O)c1 C1(NC(CCC=C)=O)COC2(CCN(Cc3cccc4cccnc34)CC2)C1 c1(C(N2CCCC(C(N3C(C)C(=O)NCC3)=O)C2)=O)ccn2ccccc12 C1(NC(c2cn(CCC=C)nn2)=O)(COC)CCCN(C(=O)C(CC)SCC)C1 C(=O)(CCC1=CCCCC1)NCC1(C(C)(C)OC)CC1.C12CCOCC1C(=O)N2 CC1=C(C(=O)Nc2cnn(C3CCN(C(=O)OC(C)(C)C)CC3)c2N)CCC1 CC(C)C(C)N=c1ccnc(N(C)CCn2ccnc2)[nH]1 n1(SCC(=O)NC(CCNC(C=C(CCC)C)=O)C)c(CC)nc2ccccc12 C(=O)(N1CCCc2nccn21)C1C(C)CCN1C(c1cccn2nccc12)=O c1(C(N2CC3(OCC(NC(CC4(C)CC4)=O)C3)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(Cc2cccc(C)c2F)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 C12(C(N3C(CNC(COC4(C)CCC4)=O)CC3)=O)CCC(N(C)C)(CC1)CC2 c1(SCC)ccccc1C(N1CCC(N(C)C(C2CCOC2C2CC2)=O)CC1)=O C1(NC(C(c2c(C)noc2C)C)=O)CC2CCC1N(C(c1n[nH]c(=N)[nH]1)=O)C2 N1(C(c2c(C)cn(C)c2)=O)CCOCCC1C(=O)NCCCc1ccco1 c1(C(=O)NCC(CC=C)NC(=O)CC=C(Cl)Cl)cc2cccc([N+](=O)[O-])c2[nH]1 N1(CC(N2CCCC2Cn2cc(CNC3CC(F)(F)C3)nn2)=O)CCCS1(=O)=O CN1CCCC12CCN(C(C1(CNC(c3cnc(=N)[nH]c3)=O)CCCO1)=O)C2 c1(C(=O)NC(CCOC)CNC(=O)CCn2cccn2)cc(Br)cnc1O C(=O)(CC(C(F)(F)F)N(C)C)N1CCC(C(N(CC(C)C#N)C2CC2)=O)C(C)(C)C1 N1(C(c2cc(OC)n[nH]2)=O)CC2CC(NC(=O)CC(F)(F)C(F)F)C(C2)C1 N1(C(c2cccc(N)c2O)=O)CCC2C(C1)CN2C(c1ccc(C2CC2)cn1)=O Cc1cc(Br)cc(C(N2CC(F)(F)CC2CCNC(C2CC2CF)=O)=O)c1N c1(Sc2c(C(=O)OCC)cc(Br)cc2SC)nc2c(Br)cccc2s1 c1(C(=O)OC)cc(NC(c2ncccc2CO)=O)cc(F)c1.C12CC3CC3N1C2=O C1(CNC(C(COC)COC)=O)CN(C(c2cc(C(F)F)cs2)=O)C(C)(C)C1 CCC(C)C(C(=O)NCCC1(NC(=O)Cc2nocc2C)CC1)NS(C)(=O)=O S(=O)(=O)(c1ccc(=NCC2CC2(Cl)Cl)[nH]c1)NCc1ccc(N(C)C)c(F)c1 N1(C(COCC(=O)NC)=O)C2CCC(C2)C1C(=O)NCC(CC1CC1)CO CCCC(C)(O)CC(=O)N1CCN(C)C(C(=O)N(C(C)C(C)C)C2CC2)C1 C(=O)(CCP(C)(C)=O)NC(CNC(C(c1ccc(Cl)cc1)C)=O)CO C1(NC(c2cc(CC)nn2C)=O)CC12CCN(C(c1occc1C)=O)CC2 c1(C(=O)NC(C2CCCN2C(C2CC3C=CC2O3)=O)C)ccc(O)nc1 C1(NC(C(C)SC)=O)CN(C(=O)COCCOCCO)CC1N(C)C CC1CN2CCN1C(C(=O)NCC(C)CNc1ccc([N+](=O)[O-])cc1)C2 C1(C(=O)NC2C(NC(CCNC(N)=O)=O)CCCC2)Cc2cncn2C(=O)N1 C(=O)(CCC(C)(C)C(=O)OC)NCC1C(NC(c2c(OC)cncc2)=O)C1 N1(C(CNC(=O)OCC)=O)CCN(CCN2CCCC2C)CC1 C(CCC(O)C(=O)NCc1nncs1)OC(C)C.C12(CC1)C(=O)NC2 C1(CNC(c2nc(C3CC3)cs2)=O)COCCN(C(c2cc(O)cc(Cl)c2)=O)C1 C#Cc1ccc(C(=O)NC(C)(C)CCCNC(c2coc(C(F)F)c2)=O)cc1F c1(C(=O)OCC)cc(Cl)cc(Cl)c1NC(=O)C(N1CCCC1C1CCOC1)=O N1(c2nccc(OCCOC)n2)CCC(NC(C2CC(=O)N2)=O)C(C)(C)C1 N1(C(CCSCC)=O)CCOC2(C1)CN(C(C1(C)CC1(F)Cl)=O)C2 c1(C(=O)NCC(C)N(C(c2cc(C)sc2C)=O)C)cccc(S(C)(=O)=O)c1 N1(C(C2(COC)CC2)=O)C2CCC1C(CO)N(C(c1csc(CC(C)C)n1)=O)C2 C1(C(=O)NCCSCC)CCN(C(=O)Cc2cccc(OC)c2)C1(C)C c1(C(=O)NCC(C)CN(C)C(C2CC2CF)=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 C(C(C(=O)NC1CCC(NC(=O)CC2COCCO2)C1)OC)OC c1(C(=O)NCC(c2ccccc2)NC(=O)CC2CCC2(F)F)ccc(O)nc1Cl CS(C)(=O)=NCC(=O)N1CCC(O)(CNC(=O)CC2CCCCC(=O)N2)C1 C#CCCCC(=O)N(CCN(C)C(c1ocnc1Br)=O)C(C)C N1(C(Cc2nc(C(C)C)sc2)=O)CCC(C2CCN(C(=O)CSC3CC3)CC2)C1 C(=O)(C(O)P(C)(C)=O)N(CCN(C(C(CC#C)O)=O)CC)CC c1(CN(CCCC)C(C2CCN(Cc3cncc(F)c3)CC2)=O)ccc(O)cn1 C1(NC(C(C)C)=O)C2CC1N(C(=O)C(=O)C1CC1)C2 C1(NC(c2ccc(Cl)cc2Cl)=O)C2COCC1CN(C(c1cc[nH]c1)=O)C2 c1(C(N2CCC(CSC)C2)C(=O)NCCC)nnc(-c2ccccc2)s1 c1(CN2C(C(=O)NCC3(C)OCCO3)CCCC2)cccc2nonc12 CCCCC(C)CCC(=O)NCC1(F)CC(NC(c2cncc(F)c2)=O)C1 C(=O)(C(CC(C)C)C(C)C)NC(CC(=O)NC(CSC)(C)CO)C(F)F C1(C(=O)NC2C=CCN(C(=O)C3=NOCC3)C2)Cc2nccn2C1 Cc1cc(C(=O)CCC(=O)NCC2(O)CN(C(C3CCCN(C)C3)=O)C2)c(C)s1 C1(C(N2CC(CC(C(=O)N(C(C)C(C)n3cccn3)CC)F)C2)=O)COCCC1C C(=O)(CC1=CCCCC1)N1CCC(C=C)(C(=O)NCC(F)(F)COC)C1 c1(OC)ccc(CN2CCC(F)(C(=O)Nc3cncc(C(F)(F)F)c3)C2)cc1I C1(C(=O)NCC2(C)CCCO2)CC2CCC(C1)N2C(c1cc(CO)on1)=O c1(C(=O)NCCN(CCC)C(C2(C)CC(C3CC3)=NO2)=O)ccnn2ccnc12 O=C1CC(C(=O)NC2CCCCC2C(=O)NC2(c3ncc[nH]3)CC2)=NN1 c1(C(N2C3C(NC(c4[nH]cc(C)c4C)=O)C(C3)C2)=O)ccc2c(c1)CCCC2 N1(C(c2c(OC)cc(OC)c(Cl)c2)=O)C2CCCC1CN(C(C1CC1C)=O)CC2 C(C1CN(C(C2(C(N)=O)CC2)=O)CC1C(=O)NC(C12CCC(CO1)C2)C)=CC C(=O)(C1c2c[nH]nc2CN1C(=O)CCC1CC1)NC1CN(CCC)C(=O)C1 Cc1csc(C(C)C(=O)NCC2CCCC2NC(c2cnc(C(C)O)s2)=O)n1 c1(C(N2CCC(c3nncn3C)CC2)C(=O)NC)ccc(F)cc1 Cc1ccc(N(CCC#N)C(=O)NC2CC(=O)N(c3ccccc3Cl)C2)cc1 N1(C(CCc2cc(C)on2)=O)CC(C(=O)NC2CC3(CCCC3)C2)C(C)(C)C1 C1(C(=O)NCC2N(C(C=CCOC)=O)CCCC2)CCn2c(C)cnc2C1 C1(NC(=O)Cn2cncn2)CCC12CCN(C(=O)COC(F)F)CC2 Cc1cc(C(N2CCSC(C(N3CC4CC4C3C#N)=O)C2)=O)cc(Cl)n1 C1(C2CCOCC2)(C(=O)NCC(CNC(=O)CCc2cc(Cl)no2)O)CC1(F)F c1(C(=O)NCC(C)(C)CNC(=O)CCNC(c2ccsc2)=O)ccc([N+](=O)[O-])o1 C=CCC(C(=O)N1CC(C)(C)C1C1CC1)NC(C1(CCC)CCCC1)=O C(C1OCCc2ccccc21)NC(C1CCN(C(c2nn(CC)c(C)c2)=O)C1)=O CCCC(C)(C)CC(=O)NC(C1(O)CCN(C(=O)CC(C)CC(C)C)C1)C C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CC2CC1N(C(C1(O)CCC1)=O)C2 C(=O)(C1Cc2ccc(Cl)cc21)NC(CNC(c1c(C)c(F)ccc1)=O)C c1(N(C(CC2(C(=O)NCC)CC2)=O)C)cc(N)ccc1SSC.C(CCCOC(=N)O)OC.O c1(-n2c(C(n3ccnc3)CC)nc(CC3CC3)n2)cc(F)ccc1F C=CCC(CNC(c1cnco1)=O)NC(C1OCCC1CC)=O C(=O)(CS(=O)(=O)N1CCC(C)CC1)NCCN(C(c1c(OC)csc1)=O)C C1(OC)CCCCC1NC(C1(C)NC(=O)NC1)c1ccccc1OC(F)(F)F c1(C(=O)NCCCC(C)NC(c2ccc(CC)[nH]2)=O)c(F)ccc(C)c1Br N1(C(C2CCC(CC)CC2)=O)CCCN(C(=O)C2=COCCC2)CC1 N1(C(c2c(C)ncs2)=O)CC(NC(c2ccc(CN(C)C)cc2)=O)CC1CO CN1CC(n2cc(C3(C)CN(C(=O)C(C4CCOCC4)=O)C3)nn2)C(O)C1 Cc1cc(S(N)(=O)=O)oc1C(N1CC2CC1CN2C(c1cnc(O)o1)=O)=O CC(C)(F)CC(=O)NCC1CC1CC(=O)NCCCCCC1CC1 N1(C(C2CN(CC)C(=O)C2)=O)CC(CC(=O)Nc2cncnc2O)CC1(C)C c1(CC)nc(C(=O)NC2CC(CNC(c3cnncc3O)=O)C2)c(N)s1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(CCN(C(c3cnn(C(C)C)c3F)=O)C2)C1 C1(C(N(CCCOCCN(C(C2(OC)CCC2)=O)C)C)=O)CCc2c[nH]nc2C1 C(CC(C)C)(C(=O)OC)N(C(c1ncc(I)s1)C(=O)NC1CC1)C CC1(C)OCCN(C(C23CCC(NC(=O)C=Cc4ccco4)(CC2)C3)=O)C1CO CC(CN1CCOCC1)C(=O)N1CC(OCCNC(C2(CCC#N)COC2)=O)C1 c1(C(=O)NCC(C)(C)NC(=O)CC2(O)CCOC2)nn(C(C)(C)C)cc1Br c1(C(=O)NCC2C(NC(c3ncc(OCC)nc3)=O)C2)cc2cccc(F)c2o1 CCC(C)C(CC(=O)N1CC(COC)CC(C)C1)NC(C1(CSC)CCC1)=O c1(OC)cccc(F)c1CN1CC2C(NC(=O)Nc3cccc(C)c3F)C2C1 Cc1c(C(=O)NC2CC(NC(C3CCCC(C(F)F)C3)=O)C2)noc1C1CC1 C1(CNC(Cn2ncc(C)c2)=O)CCC(C)CN1C(c1csc(Br)n1)=O C1(NC(C(C)O)=O)CN(C(c2c[nH]nc2-c2ccco2)=O)CCC1C Cc1ccc(-n2cncn2)c(C(=O)NCCCCCNC(C2C=CCC2)=O)c1 N1(C(CC2CCCC(C)C2)=O)CC2CC(NC(c3cnc(F)c(F)c3)=O)CC1C2 Cn1c(I)cc2c(NC(C3CC3NS(=O)(=O)CCCCCl)=O)ncnc12 c1(NC(c2ccc(-c3ccc(O)cc3O)nn2)=O)ncc(F)cc1Br C12(C(=O)NC3(CO)CCN(C(=O)Cc4ccc(Cl)c(F)c4)C3)CCCC1CCC2 N1(c2nnc(C(C)(C)C)o2)CC(NC(=O)C2=CCCCCC2)CC2(CC2)C1 CCCCC(CCCC)C(=O)NC1CC2CC(NC(c3cccc(C)c3)=O)C1C2 c1(CCNC(C(=O)NC2C(C)C2(F)F)=O)csc2ccccc12 C(=O)(C(O)CN1CCCC1)NC(C)CN(C)C(C1(C)CSC1)=O N1(C(COC2CN(C(C)=O)C2)=O)CC=C(CC(=O)N2CCCNC(=O)C2C)CC1 N1(C(c2cnc(C)s2)=O)CC2CN(C(=O)C=Cc3cnccn3)C2C1 Cc1cncnc1N1CCCC1C1CCC(N2CCC(CO)CC2)CC1.C(N)=O C(=O)(C1=CCC2CCC1N2C(C12C=CC(CC1)C2)=O)N1CC(C(=O)OC)C2(C1)CC2 C1(C)(CNC(C(C)=C(CC)C)=O)CCC(NC(c2occc2C2CC2)=O)C1 CCC(C(=O)NCc1cc(C(=O)NCC2(CC)CCOC2)no1)SC C1(NC(C2(OC)CCN(C(c3ncccc3Cl)=O)C2)=O)CCOCCC1C c1(C(=O)NC2(CNC(CN(CCOC)C)=O)CCOC2)cnn(CCO)c1C Cn1c(=N)[nH]c2cc(C(=O)NCC3(NC(=O)C=CBr)CCC3)ccc12 N1(C(CCS(=O)(=O)NC)=O)CC2(CCC2)CC1CNC(=O)CCn1cccn1 C1(C(=O)NCC(=O)NCC2C(NC(CCNC(=O)OC)=O)C2)CCCCC1 N=c1nc(C(N2CC(O)(C(F)C(=O)NCC(O)C3(Cl)CC3)C2)=O)[nH][nH]1 C(CCSC)(CN=c1[nH]c(C)cc(=NC2C=CCCC2)[nH]1)NS(CC)(=O)=O N1(C(C(C2CCCOC2)OC)=O)CCC(N(C(=O)C2=CCOC2)CCO)CC1 CC1C=C(C(=O)N2CCC(C)(CCNC(=O)C=CC3CCOCC3)C2)CC1 C#CC1CCCC(NC(=O)CCCCCN(C)C(C2(C#N)CC2(C)C)=O)C1 CCC(C)(C)C(=O)NC1CCOC1C(=O)NC1(c2noc(C)n2)CC1 Cc1ccc(S(=O)(=O)COC(CNCCc2ccccc2)C)cc1 C(=O)(N=c1c(Cl)c[nH]cc1Br)C1C2CN(c3nc(C)nc4c3ccs4)CC21 c1(CC)ccc(C(N2CC3(CC3)CC2CNC(c2occc2C)=O)=O)c(C)c1 C#Cc1cc(C(N2CC3(C2)CN(C(C2(C)COC2)=O)C3)=O)cc(N)c1 c1(OCC)cc(C(N)=O)ccc1C.c1(C2c3nnnn3C2)cc(C(C)C)n[nH]1.OC Cc1cc(C(=O)NC2(C)CCCN(Cc3nc(CN)oc3C)C2)ccc1Cl CC(C)CC(C)CC(=O)NC1CC2C(NC(c3cn4cccnc4n3)=O)C2C1 N1(C(C(C)CC2CCCC2)=O)CCC2(CCCCC2NC(C2(C)CC2C)=O)C1 C1(C(C)NC(CCc2cc(C)no2)=O)CN(C(C2(N=[N+]=[N-])CC2)=O)CCO1 C(=O)(CC(C)CNC(c1nnnn1Cc1ccco1)c1cscn1)OC N1(C(=O)COC2CC2)CC2CC(C1)N(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 CCC(F)(F)CC(=O)N1CCOCC(C(=O)NCC2(C#N)CCOCC2)C1 N1(C(c2ccc(O)cc2)=O)CCC2CN(c3ncc4[nH]ccc4n3)CCC12 c1(OC(C(=O)Nc2ncn(CCO)c2NC(=O)OC)C)ccc(F)cc1F c1(CC(=O)NC2CC(CCNC(C3C(C)(C(C)C)C3)=O)C2)c(Cl)cccc1Cl CC(C)CC(CNC(C1CCN(C(C2CC(O)C2)=O)CCO1)=O)CO C(c1csc2ccccc12)=CC(=O)NC1CCC(C)N(C(c2ccncc2)=O)C1 N1(C(c2cc(C)n(C)n2)=O)CCC(NC(=O)C(C)P(C)(C)=O)CC1C1CC1 C1(C2CN(C(=O)C(C)(C)c3ccno3)C2)(NC(C2CCC(OC)C2)=O)CC1 CCC(C)(C)CCCC(=O)N1CC(CC2(C#N)CCC2)C1 c1(CC(=O)NC2CCCC(NC(C3(O)CCOC3)=O)C2)nc2ncccn2n1 c1(CNC(C2C(C)=CCS2)=O)nnn(C)c1C(=O)NC1CCC2CCC12 C1(NC(CN(C(C)C)C)=O)COC2(CNC(Cn3ncc(CC4CC4)c3)=O)CC1C2 C1(CNC(C=CC(C)(C)NC(C2CC(=C)C2)=O)=O)CC(O)C12CCC2 C1(C)(CNC(C(=O)NCCOC)=O)CN(C(C2(Cl)CC2(F)F)=O)CCO1 C1(NC(C(C)CF)=O)CCC(C)(C)CC1CNc1cc(O)nc(O)n1 N1(Cc2ncn(C)n2)CC(NC(=O)C(=O)c2ccco2)C(O)C1 C1(CNC(COCC)=O)CC2COCC2N1C(C1CCCN1c1ncccn1)=O CCC(C#N)C(=O)N1CCC(N(C)C(c2cccc(C(=O)N(C)C3CC3)c2)=O)C1 C1(C(N(CCC(C)C)CCO)=O)CN(C(=O)C2=NOC(C)(C)C2)CCC1(C)C C(=O)(C1CCCn2cnnc21)NCC(CNC(c1cnc(CC)s1)=O)(C)C c1(C(=O)N(C2CCC23CCNCC3)CC2(C)CCC2)cc2ccc(Br)cc2[nH]1 C1(C)(C(=O)NC2(CCC)CCNC2=O)CCCN(C(=O)CCCN(C)C)C1 CCCC(C)(O)CC(=O)N1CC(CNC(=O)C(C)OC)CC1C.C1CO1 c1(NC)cc(CC(=O)NCC2(NC(c3cnn(CCN(C)C)c3)=O)CC2)ccn1 N1(C(c2c(C)cns2)=O)CCCN(C(c2ccccc2Cl)=O)CC1 N1(C(CC(C)CNC(=O)Cc2cc[nH]n2)=O)CCC(C)C(O)C1 CCS(=O)(=O)CC(=O)N1CCC(C)(NC(=O)CSc2nncn2C(C)C)C1 C(c1cccs1)=CC(N1CCCC1C1(C(N2CC(CCO)C2)=O)CC1)=O c1(C(C(=O)NCC(C)(C)OCCNC(C(C=CC)O)=O)(C)C)cc(C)ccn1 c1(C(C#C)NC(=O)CC2CCN2C(=O)C(C)CC)ccccc1 c1(C(=O)NCc2ccccc2F)cccc(CNC(c2cccc(F)c2)=O)c1 C1(C(=O)NCc2nccc(OC)c2)CN(C(=O)C(C)S(N)(=O)=O)CC1(C)C C1(NC(c2nc(C)[nH]n2)=O)(CF)CCN(C(C2(C)CSC2)=O)C1 c1(C(N2C(CNC(C3CC(OC)C3)=O)CCCC2)=O)cc(C(F)(F)F)cc(F)c1 Cc1c(C(=O)N(CCC(=O)NC(C2CCCC2)C)CCCO)cccc1O Cc1cc(CCC(N2C(C(=O)NC(C)C(=O)NC3CC3)CC2C)=O)on1 n1(CCCC)nccc1C(=O)N(CCC(C)NC(=O)C=CC(C)CC)C CCCCCC(=O)N1CC(CNC(c2cnn(C)c2Cl)=O)(OC)C1 c1(C(N2CCN(C(c3c(CC)noc3)=O)C(COC)C2)=O)ccc2cc[nH]c2c1 c1(C(C(=O)CC(C)c2ccco2)C)cnccn1.C(CCCN(C)C(C)=O)NC C12(C(N3CCC(OC)CC3)=O)CCC(C1)N(C(c1ccc(N(C)C)cc1)=O)C2 c1(C(=O)NCC=CC(N2CC(n3cnnc3)C2)=O)cc2sccc2[nH]1 N1(C(CC#N)=O)CCCC2CN(C(c3cnncc3O)=O)CCC12 c1(C(=O)NC(C2(C(=O)NC(C)C(=O)NCCF)CC2)C)cnc[nH]1 c1(NC(Cc2cccc(OCc3ccc(C)cc3)c2)=O)cnc(Cl)c(C)c1 c1(OCC)ccc2cc(C(=O)N(C(C)CNC(C3CCCN3C=O)=O)C)[nH]c2c1 N1(C(C(COC)OC)=O)CCC(NC(C2(CC(C)=O)CC2)=O)C(C)(C)C1 N1(C(c2ccc(CNC(C(C)CC3CCC3)=O)s2)=O)CC2C(C)C2C1 c1(OCC)cc(OC(N2CCN(CC(c3ccncc3)SC)CC2)=O)ccc1C C1(NC(CC(C)C)=O)CC2(CCN(Cc3ccc(O)cc3O)CC2)C1 C1(CNC(c2c(Cl)cn(C)n2)=O)CC(O)C(O)CC1C(=O)NCC12CCCC1C2 C(=O)(C(C)(C(C)C)NC(C)=O)N1C(C23CC(C2)C3)CCC1.C1(OC)(CN)CCCC1 C1(NC(=O)CC2C(NC(C3CCOC3C3CC3)=O)CC2O)CCCC(O)C1O c1(C(N2CCC(C(=O)NCCC(O)CO)C2)=O)cc2ccoc2s1 CCS(=O)(=O)CC(=O)NCC(C)NC(=O)CC(O)C1CCCC1 c1(NCc2ccc(N)c(F)c2)cc(=NCCCc2ncc[nH]2)[nH]cn1 CC(CN(C)C(c1cc2c(o1)CCCNC2=O)=O)N=c1[nH]c2cccc(F)c2s1 c1(CC)cc(CC)nc(N(CC(C)CNC(=O)CCc2cnccn2)C)n1 N1(C(CCCC=C)=O)CCN(C(c2coc3c2CCCC3)=O)C2CS(=O)(=O)CC12 c1(C(N2CC(NC(CCOC(C)C)=O)CC(C)(C)C2)=O)c[nH]c(=N)c2[nH]ccc12 N1(C(CCN(C(=O)CC2COC(=O)C2)C)=O)CC2C(C1)C2(F)F CCC1=C(C(=O)NCC(C2CC2)N(C)C(C2(F)CCCN(C)C2)=O)CCCO1 N1(C(C)=O)CC2(NC(=O)Cc3cc(OC)cc(Cl)c3)CCC1CC2 C(=O)(C1CCc2ccc(Cl)nc21)NC1(CCNC(=O)CC2CCC2)CC1 c1(C2(C(N3CCC(c4scc(C)n4)CC3)=O)CCC2)ccc(F)cc1Br CCCC(C(=O)N(C)CC1COCCN1C(c1csc(=NC)[nH]1)=O)OCC c1(C(=O)NC(c2c(OC)cccc2)Cc2ccccc2)cc(F)cc(F)c1Br c1(C(N2C(C)(CNC(C(CC)=CC)=O)CCC2)=O)nc(CC)n2ccccc12 CC1(C)NC(=O)N(CCCC(N2CC3CC2C3CNC(=O)C=CC2CC2)=O)C1=O C1(C2CCCCC2)(C(N2CCN(C(C3C(C(C)C)C3)=O)C(C3CC3)C2)=O)CC1 c1(CC(=O)NCC(CC)NC(=O)C(C)C2CCC2)ccn(CC(C)C)n1 c1(C(N2CCC(CC(C)NC(C3(C)CCCO3)=O)CC2)=O)nccc(C#N)c1F C1(O)(CCNC(Cc2cc(C)ns2)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1 C(=O)(C(C)(C)CC(F)F)N1CCC(F)(C(N(C)CC2(Cl)CCC2)=O)C1 C1(C(=O)NC(C)(C)CC2(O)CCN(C(C3CC3F)=O)CC2)C2CCC3C(C2)CC13 C=CCC(C(=O)NCC(C(C)(C)C)NC(C1CCC(=C(F)F)CC1)=O)C(C)C c1(CC(N2CC(NC(C3(Br)CC3)=O)C(O)C2)=O)c(Cl)cccc1Cl N1(C(CC2C(=O)NC(=O)N2)=O)CCC2CC2(C(N2CCn3nccc3C2)=O)CC1 c1(CN(C(CN(CC(=O)N(CCOC)CC)C)=O)C)csc(C)c1.c1(S)ccccc1 C=CC1(C(N2CCC3CC23C(=O)OC)=O)CCN(C(=O)CCC(C)=O)C1 c1(N2CC(NC(c3cnc4c[nH]nc4c3)=O)(CO)C2)nc2ncc(Cl)cc2s1 N1(C(c2ccc(C)c([N+](=O)[O-])c2)=O)CC(NC(C2(C)CC2)=O)CC12CCOCC2 c1(C(=O)NC2CC(C)(NC(c3coc(Br)c3)=O)C2)cc2nc[nH]c2cn1 C(=O)(C1CCc2ccccc21)NCC(C)(OC(F)(F)F)NC(=O)C1CC1 CC(CCCC(=O)N1CCC(F)(F)C1)NC(=O)CN1CCC(F)CC1 C(c1ccccc1)=C(C(N1CC(CCNC(C(CC)OC)=O)C1)=O)C CC1(CNC(=O)CC2CC2)CCCN(C(c2cc(C3(O)COC3)on2)=O)C1 CC(C)(C(=O)N1CCCC(CNC(C2(F)CCN(C(C)(C)C)C2)=O)C1)S(C)(=O)=O N1(CCCC(=O)NCCCN(C(C2C3CCC(=O)C23)=O)CC)C(=O)CCC1=O C1(C(=O)Nc2cn(CCC)nn2)CCC(F)(Cn2nc(C)cc2C)C1 CC(CF)CC(=O)NC1(CNC(c2cccs2)=O)CCOC1 Cc1c(O)nc2ccccc2c1C(=O)NC1CN(C(=O)CCCCN=[N+]=[N-])C1 c1(C(=O)NC(C(C)NC(CCCCNC(C)=O)=O)C(C)C)ccn(C)c(=O)c1 C1(NC(=O)C=Cc2cocn2)CCN(C(=O)C(=O)Nc2ccc(Cl)cc2)CC1O N1(C(C=C(C)C)=O)CCCN(C(=O)Cc2ccccc2C(F)(F)F)CC1C(C)C N1(C(CCOC)=O)CCN(C(C2CCN(C(C)=O)CC2)=O)CC1C(C)C c1(C(N(C)CC2(O)CN(C(C3(CCOC)CCCC3)=O)C2)=O)cc(O)ccc1F C(CC(O)C(F)(F)F)NC(C1(NC(Cn2ncc(CC)c2)=O)CC(F)C1)=O c1(NCC2N(C(C(CCC)C)=O)CCCC2)cc(C)c([N+](=O)[O-])cc1[N+](=O)[O-] Cc1ccc(F)c(CNC(Cc2ccccc2)CN)c1 c1(C(=O)NC2(CNC(C=CC(C)C)=O)CCOC2)ccc(S(N)(=O)=O)cc1F N1(C(C(C(C)C)C2CCC2)=O)CCCC(C)(C)C1C(=O)N(C(CCO)C(F)F)C N1(C(C(C)C2CC2)=O)CCC(C(=O)NCCC(C)(C)O)=C(F)C1 C1(C)(C(=O)NCCCC#C)CCN(C(c2ccc(F)c(F)c2)=O)CC1 Cc1c(Br)ccc(CNC2CC2C(N2CCOC3CC23)=O)c1F C1(NC(=O)CCF)CC(NC(=O)C=C2CCOCC2)C(O)C1 c1(C(=O)NCCN(CCC)C(C2CCOC2C(C)C)=O)cnc(NC(C)=O)o1 O=C1NCC2(CCCCC2)C1Nc1cc(Cl)cc(I)c1 N1(C(c2nccc(CC)c2)=O)CC2CC(NC(=O)C=Cc3ccco3)CC2C1 N1(C(c2ccc(NC(C)=O)c(F)c2)=O)CC2(C1)CN(C(=O)C(C)CO)CC2CO C(=O)(CC(C)(C)CN(C)C)N(C1CCN(C(=O)C(c2ccccc2OC)C)C1)C.CO N1(C(c2c(CC)onc2C)=O)CCN(C(c2cc(Cl)no2)=O)C(CCOC)C1 C(c1ccccc1OCCC(=O)NCC1CC(C)N(C(=O)CSC(F)F)C1)OC N1(C(CCCc2ccc(OC)cc2)=O)CC(NC(=O)Cc2cncs2)CC1(C)C C1(c2n(CC)nnn2)(Nc2cccc(C(F)F)c2C)CCOCCC1C N1(C(C(CCC)NC(=O)C=CC(=O)OCCNC)=O)CCCC2(C1)N=N2 N1(C(CCC(CC)OC)=O)CC2CCCC(C1)N2C(C1CC(CC)=NO1)=O C(=O)(C(C)(Cl)Cl)NCC(C)(C1CC1)NC(COCC(C)Nc1ccccc1)=O c1(C(=O)NC(CNC(CNC(CCC)=O)=O)C)ncc(N)cc1Cl O=C1CC(=O)CC(C(N2CCC2CC(=O)NCCOCC(F)(F)F)=O)C1 C1(C(N2CCC(O)(CCNC(c3c(CC)cco3)=O)C2)=O)CC2CC1CC2(F)F O=C(N=c1c(Br)c[nH]cc1Br)C1CN(C(c2ccc(B(O)O)cc2)=O)CCC1O c1(N2CCC(C(C)NC(c3ccnn3C3CC3)=O)C2)cc(Cl)nc(S(C)(=O)=O)n1 c1(CC)cc(C(N2CC(NC(=O)CCF)C(F)C2)=O)c(C)nn1 c1(C(=O)NC(C2CCCC2)CNC(C(C)SCC)=O)cccn2c(C)nnc12 C12(NC(CCC#C)=O)CCCN(C(c3ccnc(C)n3)=O)CC1C2 C1(NC(c2cccc(F)c2F)C)CCc2c(nc(Cl)n2C)C1 C(CCNC(C1CCC12CCC2)=O)(C(C)C)NC(Cc1c(C)ncs1)=O N1(C(C2CC(C)OCC2)=O)CCCC2(C1)CN(C(c1nn(C)cc1N)=O)C2 CCCCC(C)(F)C(=O)N(C1CN(C(C2CC(CF)C2)=O)C1)CC(C)C CC1(C)CCC(NC(=O)C=Cc2cocn2)C(CNC(c2ccc(Cl)[nH]2)=O)C1 c1(C(=O)NCC2(F)CN(C(COCC#C)=O)C2)cncc2ncccc12 c1(CNC(C=C(C)C)=O)cnn2c1CN(Cc1ccc(OCCO)cc1)CC2 Cc1ccc(C(F)(F)C(=O)NC(C)(C)CCNC(C2CCCS2)=O)nc1 N1(C(C2C(C(C)(C)C)C2)=O)CCCC2C(NC(C3CC3C(C)(C)C)=O)C(C)(C)C12 c1(C(N2CCN(C(C3CC4CCC3C4)=O)CC2)=O)c(F)ccc2nc[nH]c12 O=C(NNc1cc(F)ccc1F)NC1CC(c2ccc(Br)cc2)C1 N1(C(c2cccc(C(=O)OC)c2C)=O)CCn2ncc(OC)c2C1C N1(C(C2N(C)CCC2)=O)CCC2OCCN(C(=O)CC3CCCCO3)C2C1 c1(Cn2nc(CC)c(Br)c2)cnc(OC)c(C)c1 c1(C(=O)NC(C)CNC(=O)CCC(C)(F)F)cc(S(N)(=O)=O)cc(Cl)c1F N1(C(c2c(C)coc2C(C)C)=O)C(C)CC2CN(C(=O)CNC(N)=O)CC12 C1(C(=O)NC2(C(=O)NC3C(C)(C(F)F)C3)CC(CO)C2)C2CCCC1CC2 C(=O)(C(C(C)O)NC(=O)Cc1ccsc1C)NCc1c(CC)con1 CN1CCc2nc(C(=O)NCC34CCCC3CCN4C(=O)CC(F)F)sc2C1 CCC(CC)CCC(=O)NC(CNC(=O)CC(C)(C)C#N)C1CC1 CC1CCOCCN1C(C1C2CCN(C(C3C4CC5C(C4)C35)=O)CC12)=O C=C(Cl)CC(C(=O)Nc1ccc(C2CC2)nc1)NC(c1ncc(C)cc1F)=O N1(C(c2ccn(CCC)n2)=O)CCCCC(C(N2CC3CCC3(C)C2)=O)C1 Cc1ccc(C(=O)NCCCCCNC(c2cc3occc3s2)=O)c2c1CCC2 C(F)(c1ccccc1)=CC(=O)N(C1CN(C(=O)C(C#N)C2CC2)CC12CC2)C C#Cc1cncc(NC(=O)C(O)CCCNC(=O)C=CCOC)c1 CC1CCN(CC(=O)N(CC(O)CN(C)CCC2CCCN2C)C)CC1 c1(C(N2CC(C)C(NCc3cc(Cl)c(Cl)cc3F)C2)=O)cc(F)c(F)cc1F C12(C(N3CCC(C(C)(C)NC(C(C)OCCOC)=O)C3)=O)CC(CCO1)C2 c1(C(C)C)cccc(CC(=O)NCCOCCCNC(c2ccon2)=O)c1 C1(NC)CCC(CNC(=O)CCN(C(c2cc(C(C)C)[nH]n2)=O)C(C)C)CC1 c1(CC2C3CN(C(N4CCCC5(COC5)C4)=O)CC2CC3)cc(F)c(F)c(Cl)c1F C1(CCC)CN(C(C2C3CC(=O)CC23)=O)CC1CO.C1=CC(=O)NC(C)(C)C1 Cc1n[nH]c(C)c1CC(=O)NC1(CNC(=O)CCOCC(F)(F)F)CCOC1 C1(S(N)(=O)=O)(C(=O)NCCC2N(C(c3n(C)nc(O)c3)=O)CCCC2)CCCC1 c1(C(N2CC3CC(C2)N3C(c2c[nH]c3cnccc23)=O)=O)c[nH]c2ncccc12 CC1CC(CO)N1C(c1ccc(CNC(c2csc(=N)[nH]2)=O)o1)=O c1(N2CC(CC=C)(NC(=O)CCc3ccccc3F)C2)cc(C(N)=O)nc(Cl)n1 c1(OCC)cc(Br)c(C(N2CCCN(Cc3ccc(O)cc3)CC2)=O)cc1OC N1(C(CC(C)OCC2CC2)=O)CCN(C(=O)C(F)(F)c2cccnc2)CC1C S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(C3(F)CCCOC3)=O)C2)c1)N(C)C C#CC(CNC(=O)C(C)(C)NC(=O)C(CC=C)CC=C)CC(C)(C)C Cc1cc(Cl)ccc1C(=O)N(C1CCCN(C(=O)Cn2cnc(C#N)n2)C1)C c1(C(N(C(C2CCS2)=O)Cc2cccs2)=O)ccccc1 c1(NC(=O)C(N2CCC3(CCSC3)C2)=O)cccc(P2(=O)CCCC2)c1 N1(C(C)(C)C)CCCC(N=c2ccnc(N3CCCC(c4cccnc4)C3)[nH]2)C1 CC1CN(C(=O)C(O)(C2CC2)C2CC2)CCN1C(c1coc(Cl)n1)=O c1(CC)cc(C)ccc1C(N1CCCC(N(C)C(c2ccn(C)c2CC)=O)C1)=O C1(NC(c2ncc(OCC)nc2)=O)C(C)CN(C(=O)Cc2scnc2C)CC1C Cc1cc2sc(C(=O)NC3CCN(C(=O)Cn4ccnn4)C3(C)C)cc2s1 C1(C(N2CC(CO)(NC(=O)CCN3CCC3)C2)=O)(CC)CCOCC1 C1(C(N(CCOCCNC(CCSC)=O)C)=O)CCC(=O)N1C1CC1 S(=O)(=O)(c1ccc(C(N2CCC2CNC(=O)CC2(O)CCCCC2)=O)o1)NC N1(C(COC2(C)CCCC2)=O)CCC(C(=O)NCC2CCC3CC23)=C(F)C1 N1(C(C(=O)NCC)=O)CC(C)C(NC(c2ccc(C3CC3)cn2)=O)C(C)C1 C1(C(N(C(C(=O)OC)C)C2CC2)=O)CCC(c2ccc(C)cc2)CC1 c1(CNC(=O)COC2CCOC2)c[nH]nc1C(=O)NCC1CCOC1 N1(C(C(C(C)C)CN(C)C)=O)CC(NC(=O)CC=C(Cl)Cl)C2CCCC12 c1(C(C)C)cnc(O)c(C(=O)NCC(CO)NC(C2CCC2(C)CN)=O)c1 C1(C(=O)NCCCC(C)NC(CCN(C)CC)=O)CCOC(C)(C)C1 N1(c2nnc(-c3c(C)nc(NC)s3)n2CCC#N)CC(O)C(O)C12CCC2 N1(Cc2nc(C)c(C)s2)CCN(N2CCCC(c3nc(C(N)=O)cn3C)C2)CC1 CC1CN(C(c2ccc(Cl)cc2F)=O)CCC1NC(=O)Cc1ccc(O)nc1 N1(C(c2cnc(C)c(C#N)c2)=O)CC2(CCN(C(=O)Cn3cnnc3O)CC2)C1 c1(CC(C(=O)NCCCCC=C)NC(=O)C(C2CCOCC2)F)cnn(C)c1O C1(NC(CSc2n(C)nnn2)=O)C=CCN(C(c2cc(C3CC3)ccn2)=O)C1 c1(C(=O)NCC(CCOC)NC(=O)C(C)CO)cncc(N2CCOCC2)c1 C1(F)(CNC(CC2ON=C(C)C2)=O)CC2CCC(C1)N2C(=O)Cc1cccnc1 c1(C(=O)NCC2CN(C(C(COC)C)=O)CC2O)cc(F)cc2cccnc12 C(=O)(C(O)N1CCCO1)NC(C(C)N(CCO)Cc1cccc(OC)c1)=O Cc1ccc(C(N2CCC(NC(c3oc(Br)nc3C)=O)C(F)C2)=O)cc1Br C1(CC(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC2F)CC(c2ccccc2)=NO1 C=CCC(C(=O)NC1CC(NC(c2cnc(OC)c(C)n2)=O)C(O)C1)C(C)C C1(NC(=O)CCC2CCC2)COCCN(C(=O)C(O)Cc2ccc(F)cc2)C1 CC1=C(C)CC(C(=O)NC2COCC2C(=O)NCC2(O)CC2)CC1 CC1CN(C(C2C3CCC2CC3)=O)CCC1NC(C1(n2cccn2)CC1)=O c1(CN2CC(C(=O)Nc3ccc(CCC)cc3)SCC2)ccc(I)cc1Br C(=O)(CC(O)C(C)(C)C)N(CC(C)NC(c1ccc(OCC)cc1)=O)C CC1CN(C(c2ccc(Cl)s2)=O)CC(C(=O)NCCc2ccon2)O1 C1(C2CCCOC2)CC1.N1(C(C=C2CCN(C(=O)C=CCBr)CC2)=O)C2COCC1C2 N1(C(CCC2CCCCN(C(CSCCC)=O)C2)=O)CC(C)NC(=O)C12CC2 c1(C(=O)OC)ccc(OC)cc1C(=O)NC1CCCCN(C(=O)CC2(CO)CC2)C1 c1(C(=O)NCCC2(C(=O)NCc3cnc[nH]3)CCCC2)cc(F)cc(F)c1 C(=O)(CCCCC(F)F)N1CC(CNC(C2(C#C)CC2)=O)N(C)CC1 CCCCC(F)C(=O)NCCOCCCN(C(=O)C(C)(F)c1ccon1)C C(CCC(C)C(=O)N1CCC1C(=O)NC1CCS(=O)(=O)C1)OC(C)=O CC1CC=CCC1C(N1CC(OC2CCN(C(=O)C(=O)NCC(F)F)CC2)C1)=O c1(C(N2CC(NC(CCOCC#C)=O)C(C)C2)=O)cnc2n1CCC(C)C2 CC1(C)CC(=O)NCC1CN(C(=O)Cc1cccn1C1CCCC1)C1CC1 C1(C(N(C2CCN(C(CCC=CCC=C)=O)C2)C)=O)CC2(CCC2OC)C1 C1(NC(C)=O)(CO)CCCN(C(C)C(=O)NCC(C)CC(F)(F)F)C1 C(C(O)C(=O)NC(c1cnn(C)c1)C(=O)NC1CCOC1)=CCCC C(=O)(C(C)C(F)(F)C(F)F)N1CCC(N(C(C2(C)CCNC(=O)C2)=O)CC)CC1 C1(C(=O)NC(N(C)C)=O)Cc2ccccc2O1.C1(COC(C)(C)C)CC1NC=O c1(C(N(CCC(C)NC(C(CC)C(C)C)=O)C)=O)ccc2c(c1)NC(=O)CS2 CC1OCCCC1C(=O)NC1CC(CNC(=O)C=CCOc2ccccc2)C1 c1(C(C)C)ncc(Cl)c(C(=O)NC2CC23CC(NC(c2ncncc2Cl)=O)C3)n1 C1(C(N(C(C(C)C)CO)C)=O)CN(C(C2COCCO2)=O)CC1(C)C c1(C(c2n(CCC)nnn2)(C)NC2CC(O)(COC)C2)ncc(Cl)cc1F c1(C(=O)NC2C(NC(C(C(CC)C)O)=O)CCC2)cc(F)c(F)cc1OC Cc1[nH]c(C(N2CCCC(C)CC2)=O)c(C)c1C(=O)NCc1csc(C#N)c1 C#Cc1cnc(N(C)CC2CCCN2C(c2cccc(Cl)c2OC)=O)nc1 C1(O)(C(=O)NC2CC(N(C(C=CCN(C)CC)=O)C)C2)CCc2ccccc2C1 N1(C(C2C(CCC)C2)=O)CCC1C(=O)NC1(CC(=O)OC)CC1 C1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)CCN(CCO)C(=O)C1 C1(c2ccc(CNC3C(NC(=O)Cc4nn[nH]n4)C3)cc2)CCCCC(=O)N1 C(=O)(C(C)C(C)S(C)(=O)=O)N(CCCNC(C(CC)(C)C)=O)C C(=O)(CN1C(=O)COc2ccccc21)N1CCC(C)(CNC(CCCSC)=O)C1 c1(OC)ccc(CCC(N2CCC(=O)CC2C(F)(F)F)=O)c(Cl)n1 c1(NC(CN(CC(C)C)C(=O)CN(c2ccccc2F)C)=O)ccc2nccn2n1 N1(C(c2sncc2Br)C(=O)NCCOC)CCc2c(c(C3CCCO3)nn2C)C1 N1(C(CC=C)=O)CCC(NC(c2cc(O)n(CC)n2)=O)CC1 c1(C(=O)NCCC2CCCN(C(c3cnc(C)s3)=O)C2)noc2ccccc12 N1(C(c2c(C)nc(C)s2)=O)CC2OCC(NC(=O)CCOCC(F)F)C2C1 c1(C(=O)NC(C(C)(C)C)CNC(=O)CC2COC(=O)C2)cc(N)c(Cl)c(O)c1 Cc1cc2cc(C(=O)NCC3CC(C)(C)CN3C(=O)CCC(F)F)oc2cc1C c1(C(N2CC(O)(CCNC(C(CCC)OC)=O)C2)=O)c(N)ccc(Br)c1F C1(C(C)(C)O)(CNC(c2ccnn2C2CC2)=O)CN(C(=O)CC2CC(F)(F)C2)C1 c1(NC)cnc(Cl)cc1C(=O)OCC1CCC(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(C2CN(C(c3cn(CC)nn3)=O)C2)C)onc(OC)c1Br O(C1CCCc2ccccc21)C(C(N)Cc1cccc(Br)c1)=O N1(C(COc2cccc(C)c2)=O)CCC(C)C(NC(=O)C(C)(F)F)C1C CC1CC(NC(=O)CCCn2ccnc2)CN1C(=O)CCn1cccn1 C1(CCCNC(c2cc(O)ncn2)=O)CN(C(C2CC2c2ccccn2)=O)CCO1 c1(-c2n(C3C(C)(C)OCC3)nc(C3CCCO3)n2)cc2n(n1)CCCCO2 Nc1ncc(C(=O)Nc2csc3ncnc(O)c23)cc1[N+](=O)[O-] C1(C(N2CCN(C(=O)NC(c3cnccc3Cl)=O)CC2)=O)CNC(=O)CC1(C)C CC(C(=O)NCCC1(O)CCN(C(C2(c3ccno3)CC2)=O)C1)C(F)(F)F C1(OC)(CNC(c2ccc(C)c(Cl)c2)=O)CCN(C(c2c[nH]c(Br)c2)=O)CC1 c1(NCc2cc(C)sc2Br)ccc(C)c(Br)c1 C12(C(=O)NC3CCN(C(C=CCC)=O)CC3(C)C)CC3CC(C(=O)N1)C2C3 C=CC(C)(O)CC(=O)NCC1CCN(C(=O)C(=O)NCCC(N)=O)C(C)C1 c1(C(=O)NC(CCCNC(CCN(CCC)C)=O)C)ncnc(C)c1OC C(N=c1[nH]c(Cl)ncc1F)C1N(C(c2cnc(COC)s2)=O)CCCC1 CC(CSC(F)(F)F)C(=O)NC1CC(C)(NC(=O)C(Cl)=CCl)C1 CC1(C)CC(CC(N2CCCC(CCO)C2)=O)N(C(c2csc(CO)n2)=O)C1 c1(C(=O)NCC2N(C(C(C(C)C)n3ncc(C)c3)=O)CCC2)cc(O)nc(Cl)c1 C1(OC)CC2(C1)CC2NC(=O)CCN(C(c1csc(O)n1)=O)CC1CC1 N1(C(c2nc(C)sc2C)=O)CCCN(C(=O)CCOc2ccccc2Cl)C(C)C1 C1(N(C(C2C(C=C)C2)=O)C)CCC(NC(=O)C(c2ccc(OC)cc2)C)CC1 C1(OC)CCCN(C(C2C3CC2N(C(=O)C(F)F)C3)=O)CC1 Cc1cc(Br)cc2[nH]c(C(=O)NC3CC3CNC(c3ccnc(O)c3)=O)cc12 C(c1cccnc1C)=CC(=O)NC1CCN(C(CN(C)CC)=O)C1C1CC1 Cc1ncc(CC(=O)NCC2(C(=O)NCC3CCC(C(C)C)CC3)CC2)c(O)n1 CC1(C)CCC1C(=O)NC1COCC1NC(c1nscc1Br)=O N1(C(CCCOC(C)=O)=O)CCCN(C(c2cc3n(n2)CCOC3)=O)C(C)C1 C=CCC(CO)NC(=O)C(c1cn(C)nn1)NC(c1cnn[nH]1)=O c1(C(N2CCC(c3nc(C)on3)C2)C(=O)NCCCF)ccc(Cl)cc1O CN=c1[nH]cc(C(N2CCCC(N(C(=O)CNS(=O)(=O)NC)C)C2)=O)s1 C(=O)(C1=NOC(CNC(c2coc(C(F)F)c2)=O)C1)N1C(C(N(C)C)=O)CCC1 CC(C)CC(C)CC(=O)N1CCC(C(C)C(=O)NCC(n2cccn2)C)C1 Cc1onc(CO)c1C(N1CCC(NC(c2nnc(C(C)(C)C)s2)=O)C1)=O C1(C)(C(=O)NCC2(CNC(c3cn(CCC)nc3)=O)CC2(F)F)CCCC1O C1(NC(c2csc(C)c2C2CC2)=O)COC2C(NC(=O)C(C)(C)N(C)C)COC12 c1(NC(CSCCC(C)C)=O)nc(NC(=O)Cn2ccc(C(F)(F)F)n2)cs1 CC1CCCCC1OCC(=O)NCC1CN(C(c2cnc(C(F)F)nc2)=O)C1 c1(C(N2C(C)(COC)CC(NC(=O)CNC3CC3)C2)=O)ccn2cccc2c1 C1(C(N(CCCNC(C2COC(=O)O2)=O)C(C)C)=O)CC12CCOCC2 N1(C(CCOCC(C)C)=O)CCC(CC(N2CCCC2n2ccnc2)=O)C1 C1(CNC(CCSC)=O)CC(C)N(C(=O)CNC(c2cccc(F)c2)=O)C1 C(CC(CO)NC(=O)CCCN(C(=O)CCCn1cccc1)C(C)C)SC CCC(C)CCCCC(=O)NCCC(C)NC(c1ccc(-c2ccncc2)s1)=O C1(CN(C)C)CCOC(C)(C)C1.C1CC(=O)NCC2(CC2)C(=O)N1C(C)C C1(C)(C(=O)NCC(C)NC(c2ncsc2C2CC2)=O)CCC(=O)CC1 c1(C(N2C(C(=O)NCc3cc(OC)no3)C(C)CC2)=O)cc2ccccc2o1 N1(C(CC2C3CN(C(Cc4c(C)noc4C)=O)CC32)=O)CC(C)OC(C)(C)C1 C1(CNC(C2(C)C=CCCC2)=O)CN(C(=O)CCC(CF)CF)CC12CCC2 c1(C(=O)NCCCN(C(=O)CC2CCSCC2)C)cc(Cl)c(F)cc1[N+](=O)[O-] N1(C(C(C(CC)O)C)=O)CC2CCOC2(CNC(=O)CCn2ccccc2=O)C1 CN1C(=O)CC(O)(CNC(=O)COc2ccccc2)C1=O C1(NC(C2C(SC)CC2)=O)(CNC(C2COCC(C)O2)=O)CCCCCC1 c1(C(=O)NCCN(C(=O)C(C)(F)C(=O)OC)CCC)cc(C)cc(C)c1 N1(C(C=CSC)=O)CC2(CC(NC(C3CCCCCS3(=O)=O)=O)CO2)C1 C1(C(=O)NCc2cccc(C(=O)NCC3(CO)CCN(C)C3)n2)CCC(O)CN1C C(=O)(C1=C(Cl)CCCC1)NCC(C(C(C)C)C)NC(c1cc(O)ccc1F)=O CCC(C)(C)C(C(=O)N1CC2(CNC(c3ocnc3C)=O)CC1CO2)OC c1(CCN(C(=O)OC(C)(C)C)C2CC2)noc(-c2ccccc2)n1 n1(CC(=O)N(C)CC2CN(C(=O)COCC(F)F)C2)cnccc1=O CC(C)(CC(=O)NCC1(C)CCCC1NC(=O)C=Cc1cocn1)C(F)F c1(C(=O)NCC(C)(C)NC(C=CCC)=O)cc[nH]c(=N)c1 C1(NC(c2sc(C)c(O)n2)=O)C(C)CCN(C(c2ccc(C)n2C)=O)C1C C1(N(C(CCCOCCC)=O)C)CCN(C(=O)CC2(C(=O)OC)CCC2)CC1 C(CC(C)(C)C)(C(=O)Nc1cn(C)nc1O)NC(C(C(CC)C)=O)=O c1(CC(N2C(C(=O)NCc3ncc(C)s3)COCC2)=O)ccc(S(C)(=O)=O)cc1 C1(C(N2CCC(O)C(CO)C2)=O)(CC)CCN(C(c2cc(OC)ncn2)=O)CC1 c1(OC)cnc(C(=O)NCC23CC2CN(C(=O)C2=CCCCC2)C3)c(OC)n1 Cc1ccc2c(CN3CCC(NC(c4ccc(Cl)c(C)c4)=O)C(F)C3)c[nH]c2c1 C12(NC(c3coc4c3CCCC4)=O)CCC(CN(C(=O)C(F)C3CCC3)C1)C2 C1(C(N(CC)Cc2cn[nH]c2)=O)CC(NC(c2ccc(C(C)C)cc2)=O)C(O)C1 n1(CCC(C)(C)SCC)c(N2CCCC2)nnc1-c1ccc(C(N)=O)cc1 C1(C(N2CCCC(CC)C2)=O)CN(C)CCN1C(c1nc(Cl)oc1C)=O C1(CCNC(=O)Cn2cc(C3CC3)cn2)CSCCN1C(=O)COC1CC=CC1 CC(CC1=CCCCC1)NC(C1(NC(C2CC2c2ccsc2)=O)CC1)=O C#CCC(C(=O)NCC(c1ccccc1F)NC(=O)CCc1cccnc1)C1CC1 c1(C(N2CC(CC(C)NC(c3oc(CO)cc3C)=O)C2)=O)c(C)ccc(C)c1C C1(CNC(CC(CCCC)O)=O)CCN(C(=O)C(C2CC2)C2CC2)CCC1(F)F N1(C(C(C)(C)OC(C)=O)=O)CCOC(C(C)NC(=O)C(CO)c2ccccc2)C1 c1(CNC2N(c3c4cn(C)nc4ncn3)CCCC2)cc(Br)cc([N+](=O)[O-])c1 N(C1CCc2ccc(Br)cc21)C(C1CCCCN1Cc1c(Br)cncc1Br)=O Cc1nc(C2C(C(=O)NC34CC(NC(c5cn[nH]c5)=O)(C3)C4)C2(C)C)n[nH]1 N1(C(C2CCN(C(N)=O)CC2)=O)CC2(CC(NC(=O)C3=CCCO3)CO2)C1 C1(CC)CN(C(C2CC(=O)CS2)=O)CC1C(=O)NCC1([Si](C)(C)C)CC1 c1(C(=O)NC2CN(C(C(CSC)C)=O)CC(O)C2)ccc2nc(O)sc2c1 C1(F)(CNC(c2cc[n+]([O-])cc2)=O)CCN(C(c2cscn2)=O)CC1 C1(NC(=O)Cc2cnoc2)COC2CN(C(C3CCCOCC3)=O)CC12 Cc1cc(CNC(=O)COC2CN(C(c3cncc(CO)c3)=O)C2)ccc1F Cc1[nH]nc(C(N2CCC(C(C)C(=O)N(CC(C)O)C3CC3)CC2)=O)c1O c1(C(N(CC(=O)N(C2CC2C)C)CCOC)=O)cn(C2CC2)cn1 C(=O)(CC1=NNC(=O)C1)NC1(C)CCCN(C(=O)CC2CCC3(CC2)CC3)C1 c1(Cn2ncc(C(=O)NCCN(C(=O)CCCF)CCC)c2)ccccc1F c1(NC(CC2N(C(CCOCCOC)=O)CC2)=O)cccc(Cl)c1C Cc1nn(CC(N2CC3CC3(CNC(=O)C(=O)C3CCCC3)C2)=O)c(C)c1Br C1(C(C)C)COCCN(C(C2CCN2C(=O)C(F)=CC2CC2)=O)C1 C1(CCNC(=O)Cc2cncc(O)c2)CN(C(C2CC2F)=O)CCS1(=O)=O C(C(C)(C)CC(=O)NC12CCN(C(=O)CN3CCC(O)CC3)CC1C2)OC c1(C(=O)NC(CNC(c2cc(C)nc(O)n2)=O)C)ccc2c(c1)CN(C)CC2 C1(C(=O)NC2CCC3CCN(C(CCCOC)=O)C32)CCc2nc(=N)[nH]cc2C1 c1(C(N2CCC(C)(CNC(C3(NC(C)C)CC3)=O)C2)=O)c(F)cccc1F C1(C(=O)NC(CC)COC)CCOC1CNC(c1c[nH]nc1Cl)=O c1(C(N2C(C)CC(NC(=O)CCC#N)C2)=O)cnc2[nH]cnc2c1 c1(C(=O)NCCCN(C(=O)CC(=O)NC2CC2)CC)coc2cc(C)ccc12 C1(C2CCN(C(c3cn(CCCC#N)nn3)=O)C2)(NC(CC(CC)C)=O)CC1 c1(C(c2nnnn2CCC)NC2(CCCC)CCCC2)cc(F)ccc1C(F)F c1(C(=O)NN2CCN(Cc3ccc(CC)cc3)CC2)ccc(C)c(S(N)(=O)=O)c1 c1(SC)ccc2cc(C(=O)NC3CC3NC(C3OCC4CCCC34)=O)[nH]c2c1 c1(C(N2CC(N(C(CC3C(C)C3)=O)CCO)C2)=O)nc(N)cc2ccccc12 N1(C(CCc2onc(CC)n2)=O)CCCN(C(C2COCC2CF)=O)CC1CO c1(C(=O)NCC(CC(C)C)NC(C2C3CC4C(C3)C24)=O)ccc([N+](=O)[O-])n1C C1(C)(C(N(CCCCCCNC(c2c(C)snn2)=O)C)=O)CCOC(C)C1 c1(CNC(C2N(C(C(CC)N(C)C)=O)CC(OC)C2)=O)ccnc(F)c1 c1(CNC(C2CC(CNC(C3(F)CC3)=O)C2)=O)ccc2c(c1)CC2 N1(C(CC(C)C)=O)CCC(C2(O)CC(NC(C34CC(C)(CO3)C4)=O)C2)CC1 C1(C(=O)OC(C)(C)C)(CO)CCCN1C(=O)CC(=O)NCCF.CC1C(=O)N1 C1(CNC(c2csc(F)c2)=O)CC2(CC2)CN1C(c1cc(Cl)ccn1)=O C(C)(N=c1ccc2c([nH]1)CCC2=O)C1CCN(C(c2n(CCC)ccc2)=O)C1 C(N=c1[nH]n(C)cc1OC)c1cc(C(CC)CC)no1 Cc1cc(C(N2C3CN(Cc4ccc(-c5cccc(F)c5)cc4)CC23)=O)c(C)[nH]1 N1(C(c2c(CC)ncs2)=O)CCC(NC(c2cc(C)c(F)cn2)=O)C(CO)CC1 Cn1cc(C(N2CCC(CO)C(NC(=O)CC3(O)CCC3)C2)=O)c(O)nc1=O c1(CNC(=O)NC2CCN(S(CC#N)(=O)=O)CC2)noc2c1CCCCC2 c1(OCC(=O)NC(C)(CNC(=O)C=CBr)C2CCC2)ccc(CO)cc1 Cc1sc(=O)n(CC(N2CC(NC(c3nc(=O)n(C)[nH]3)=O)C3(CC3)C2)=O)c1C c1(C(=O)NC(CCN(C(c2cccc(C(C)=O)c2)=O)C)C)ccc(N=[N+]=[N-])cc1 N1(C(C(C)O)=O)Cc2ccccc2C(CCN(C)C(c2ccc(CO)cc2)=O)C1 C1(CC(N2C(C(C)NC(C3CC(F)(CO)C3)=O)CCC2)=O)CCC(F)(F)CC1 N1(C(CCc2onc(C)n2)=O)CCC(O)(CNC(c2ccc(N)c(F)n2)=O)CC1 C(=O)(C1=NOC(C)C1)N1CCC(CC#C)(C(=O)Nc2ccc(F)c(C)c2)C1 c1(NC(C2C(c3onc(COC)n3)C2)=O)cc(OC)c(Cl)cc1OCC N1(C(CCC(=O)NCCC)=O)CC(NC(=O)CN(c2ccccc2)C)CCC1C c1(C(C)(F)C(=O)NCC(C2CC2)NC(=O)Cn2cncn2)ccc(F)c(F)c1 CCCC(C)(C)C(=O)N1CCC(CCC(=O)NC(C)CN(C)C(C)C)C1 c1(C(N2CCC(N(C)C(c3snc(O)c3Cl)=O)C2)=O)nnn2c1C(=O)NCC2 C(=O)(C1CCC(=O)c2cccn21)NCC1N(C(c2cn(C)nc2)=O)CCCC1 c1(C(C)NC(=O)NCCCC(O)CO)ccc(OCC(F)(F)F)cc1F C1(C(=O)NCC(CNC(c2c(N)snn2)=O)F)CC2CCC(C1)O2 C1(F)(C(N2CCC(OCC=C)C2)=O)CCCN(C(=O)CN(C2CCCC2)C)C1 N1(C(Cc2cc(C)sc2)=O)CCOCC(NC(c2c(C)nn(C(C)C)c2Cl)=O)C1 C1(NC(=O)CN2CCCC2=O)CN(C(C2CCSCC2)=O)C2CC12 N1(C(C2(C)C(C)(C)C2)=O)CCOC(CC(N2CCC(C(N)=O)C2)=O)C1 N1(C(C2C3CN(C(C(C)SCCCC)=O)C2C3)=O)CCCN(C)CC1C N1(C(=O)CC2(OC)CCC2)Cc2ccc(NC(=O)C(=O)OC(C)=O)cc2C1 Cc1ccsc1CC(=O)NCC=CCNC(=O)C(CO)N1CCCCC1 c1(C(=O)NC2CC(CC(=O)Nc3nc(Br)cs3)C2)ccc(F)cn1 CCCCCC(C)CC(=O)N1CC2(CC(CC(=O)NCCC(C)SC)C2)C1 c1(NC(=O)NCc2cccc(C(F)F)c2)cc2ccccc2c(=O)o1 C1(C(=O)NCC(C)Cc2cn[nH]c2)CCC(O)CN1C(c1ccn(C(F)F)n1)=O c1(C(=O)NC2C(N(CCC(=O)NCc3ccccc3)C)C2)cc2ccccc2o1 c1(Cc2onc(C(C)C)n2)ccccc1S(=O)(=O)N1CCC(C(=O)O)C1 c1(C(N2C(C)(CC(=O)N(C3CC(C(N)=O)C3)C)CC2)=O)cnn2ccccc12 N1(C(C(CC=C)(F)F)=O)CC2(C1)CN(C(=O)C1=CCC1)CC(C)(C)O2 c1(C(=O)OCCC(CCC(=O)OC)C)cn2c(n1)CCCC2C C1(CNC(c2cc(C)ns2)=O)CN(C(c2cc3ccsc3s2)=O)C2(CCC2)C1 N(C(=NCc1cc(C(C)(C)C)on1)N1CCC(COC)C1)C(CC)C CCCC(C)(O)C(=O)N1CC(N(C(=O)CCc2ccccn2)CC)C(C)(C)C1 c1([SH](C)NCC2CC2(Cl)Cl)c(C(=O)O)oc2ccccc12 N(C(=NCC(Cl)C(F)(F)F)NCc1ccnc(N2CCOCC2)c1)CC1(C)CC1 C1(C(=O)NCC(C)(C2CC2)NC(C2CC23CCCC3)=O)CCC2(CCC2)CC1 Cc1ccc2c(C(N3CC4CN(C(=O)C=CS(C)=O)CCC34)=O)ccnc2c1Cl N1(C(C2C(C)C2)=O)CCC(C(=O)NCC(c2ccccn2)C)(CO)CC1 c1(C(N(C(CNC(C2CC(C(=O)OC)C2)=O)C)C2CC2)=O)cn(C)cn1 N1(C(N)=O)CCC(C(N2CC(C(=O)NCC3(N(C)C)CC3)C3CC23)=O)CC1 C1(C)(NC(C(C)C2CCCO2)=O)CN(C(C2CC3CC3C2)=O)C1 C=CC(C)(CCOC)C(=O)N1CCN(CCCNC(=O)CCC(C)SC)CC1 N1(C(c2ccc(CC)[nH]2)=O)CC(NC(=O)C(C)CC(C)CC)CC12CCOCC2 O=C(C1=Cc2ccccc2C1)NCC(CC1CC1)C(=O)NCCc1csnn1 C=CC1OCCC1C(N1CCCCC1C1(NC(C2CCC2OC)=O)CC1)=O C1(C(N2CCCC(NC(Cc3c(C)non3)=O)CC2)=O)CCn2c(O)nnc2C1 N1(Cc2c(OC(C(=O)OC)C)ccc(Br)c2)CC(C)(C)C1C1CCCO1 N12CCCC(C1)C2=O.C(CNC(c1nn[nH]c1Cl)=O)(C(C)C)NC(CC)=O N1(C(c2cccc(CC)n2)=O)CC2CC(NC(c3ncc(Cl)s3)=O)CC1C2 c1(C(=O)NCC=CCNC(=O)Cc2cccnc2)cnc(Cl)c(Cl)c1 C1(C(N(C)Cc2c(OC)cccc2)=O)CC2OCCC2N(C(=O)C=CCBr)C1 c1(C(=O)NC(CNC(COCCC#C)=O)C2CC2)cn2c(n1)COCC2 C=Cc1cnn(C)c1C(=O)NCC1CCCCC1NC(=O)CCCC(=O)N(C)C CCC(CC)CCCC(=O)N1CC2OCC(NC(=O)CCc3cncn3C)C2C1 c1(C(N(C2CCN(C(C3(CO)CC3)=O)C2C(C)(C)C)C)=O)cc2c(s1)CCSC2 C#Cc1cc(C(N2CC(NC(c3ccnn3C=C)=O)CC2C)=O)cc(Br)c1 C(=O)(CCC(=O)NN(C)C)N(CC(=O)NCCCCC1CC1)CC=C C(=O)(CCCCCN=[N+]=[N-])NC1CC=C(C(=O)NC(C)CN2CCCC2)C1 Cc1ncc2n1CCN(C(=O)C(CNC(=O)CC1CC(=O)NC1=O)CC(C)C)C2 C(CCC(C)(C)C(=O)N(CCCN(C)C)C)NC(c1c(CC)cccc1)=O c1(C(N(CC(CNC(C2CCN(CC)C2)=O)C)C)=O)cc(OC)cc(Cl)c1 N1(C(c2c(OC)cccn2)=O)CCN(C(=O)Cc2ccccc2Cl)C(CO)C1 N1(C(=O)NC(C)C)CCOC(C(=O)N(CC#N)Cc2ccsc2)C1 C1(CC(N2CC3CC(O)CC2C3)=O)Oc2cc(F)ccc2NC1=O c1(OC)cccc2sc(C(N3CCN(C)C4CC34)=O)nc12 Cc1ccn2cnc(C(N3CC4C(CNC(=O)C(C)CC(N)=O)C4C3)=O)c2c1 c1(C(NOC(C(=O)NC(CC(=O)NC)C2CC2)(C)C)=O)ccccc1C(C)OC C1(N(C2CC(C#N)C2)C(C)=O)CC12CCN(C(c1ccc(F)c(O)c1F)=O)CC2 C1(CC)(CNC(C2CCCC2NC(c2cc(Cl)n(C)n2)=O)=O)CCC(=O)N1 CCCC(CCCNC(=O)CNC(=O)CCC(CC)OC)NC(=O)CCC1CC1 Cc1ccc(C(=O)N(C2(CC(=O)N(C)CC3CC3(F)F)CC2)C)cc1O C1(F)(CNC(c2c(COC)cco2)=O)CCC(CNC(C2(C(N)=O)CC2)=O)C1 N1(C(C2CCN(C)C2)=O)CCC2(CCC(CNC(=O)CC(C)(C)C)CC2)CC1 N1(C(=O)COC2CCCOC2)CCCC(C2CCCCN2C(=O)C=CC2CC2)C1 C1(NC(C2(N(C)C)CC2)=O)CCCC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1 O(NC(=O)C(c1cn(C)nn1)NC(c1ccn(CC)n1)=O)C(C=C)C C(=O)(C#CC1CCOC1)N(CC(C(=O)NC1(CC#C)CC1)C)C N1(C(C(CC)N(C(=O)CC2(O)CCC2)C)=O)CCOC(C)(COC)C1 Cc1ccc(F)cc1C(N1CCCCCC1C(=O)NC(CO)C1(C)CC1)=O c1(C(N2CC(OC)(CNC(c3cc4ccsc4s3)=O)C2)=O)cccn2ncnc12 Cc1nn2cc(CC(=O)NC3(C4CCN(C(=O)C(O)C5CC5)C4)CC3)nc2s1 c1(C(N(CCNC(Cc2cc(C)sc2)=O)C(C)C)=O)ccc(F)c2ccsc12 c1(C(=O)NC(C=C)CO)ccc(CNC(=O)C=CC2(C)COC2)cn1 C(=O)(C(CN=[N+]=[N-])NC(=O)Cc1ccns1)NCCC1CCC(C)(C)C1 C12CCC(CC1)C(=O)C2=O.C1(OCC)CC(N)C1.C(=O)(C(C)c1ccsc1)N N1(C(CCC(C)OC)=O)CCC(F)(C(=O)NCC(C)C(O)C(C)C)CC1 CCCCCC(C)(C)C(=O)NCC1CCCN1Cc1scnc1C N1(C(C=NOC)=O)CC2CN(C(c3cc4cccnc4[nH]3)=O)CC2(C)C1 c1(C(N(CCC(=O)NCc2nncs2)C)=O)cccc[n+]1[O-] CC1CN(C(=O)COc2ccc(F)nc2)CCC1CNC(=O)CC1CCCC1 Cc1cc(Br)cc(C)c1C(N1CCC(NC(C2(n3cc(Br)cn3)CC2)=O)CC1)=O C(=O)(C(CO)C(F)(F)F)N(C1CCCCC1)CCNC(C1(C)CCC(=O)C1)=O N1(C(CCCOC)=O)CCC(C2OCCCC2NC(=O)Cc2cnsc2)CC1 c1(OC)cc(C(=O)NCC=CCNC(C2CCOC2c2ncc[nH]2)=O)sc1Cl CC#CCC(C(=O)NC)NC(=O)CCSC(C)C(=O)NC(C)C C(=O)(CCCC(=O)N1CC(N(C)C(C2(C)CC2(F)Cl)=O)C1)NCC C1(NC(C2(C)CCSCC2)=O)CC2CCC1N(C(=O)C#CC1CCOC1)C2 c1(C(=O)NC2CN(C(c3ncc(CC)cn3)=O)CC2SC)cn2cc(C)sc2n1 c1(C(N2C(CC)CN(C(C3CCC(=O)N3)=O)CC2)=O)cc2cc(C)ccc2o1 c1(CC)cc(C(=O)N(C2C3CN(C(C4CCCC4O)=O)CC23)C)cc(N)c1 c1(C(=O)NCC2CC(NC(C(COC)C)=O)C2)c(C(F)(F)Cl)n[nH]c1C C(C(=O)N1CC(N(C(=O)COc2cc(C)on2)C)C(C)(C)C1)(C(C)(C)C)SC N1(C(CCC)=O)CC2(CCN2C(c2cnc(C)c(C)c2)=O)C1 c1(C(N(CCCCNC(c2ccc(CCCCC)o2)=O)C)=O)cc(F)n(C)n1 c1(CC)cc(NC(=O)C(c2cccnc2)NC(C2CC2[N+](=O)[O-])=O)cc(O)c1 CCC1c2ccccc2CN1N1CC2(CC)CCC2(CO)C1 CC1(CNC(c2ccnc(CNc3cccc(CO)c3)c2)=O)CCCCCC1 c1(C(N(CC(C)CNC(=O)C(=O)C(C)(C)C)C)=O)ccc(N=[N+]=[N-])cc1 C1(CC(=O)NC2(C)CCS2)CN(C(C2C(Cl)(C(=O)OC)C2)=O)CCO1 C(=O)(C1=CC2C=CC1C2)N1CCCC(CN(C(=O)CC2COCCN2C)C)C1 CCC(C(=O)OC)C(=O)NC1CC(O)C1CC(N1CCCC(C(C)OC)C1)=O N1(C(C(=O)N(C(C)C)C(C)C)=O)CCCC(Cc2cc(C(C)(C)C)on2)C1 C1(CC(N2CC3CC2CS3)C(=O)NC2COC2)CCCCCC1 c1(CSC)ccc(N(C)C(C2CCC(CNC(c3nc(O)sc3C)=O)C2)=O)cc1 c1(C(=O)NC2(CCC)CCCN(C(=O)C(F)C(C)C)C2)cc2c(C)sc(C)c2s1 C1(NC(C=CC)=O)CC1C1CCCN(C(=O)Cc2nccc(OCC)c2OC)C1 c1(C(=O)NCC(c2ccc(C(C)(C)C)cc2)C)ccc(Cl)c(C(=O)O)c1Cl N1(C(c2c(C(C)C)ocn2)=O)CC2CCC2(CC(=O)NC2(C(C)(C)C)CCC2)C1 c1(NC(=O)CC2CC23CC3)ccc(S(=O)(=O)Nc2ccccc2)cc1 Cc1nn2cccnc2c1C(=O)NC1CC(NC(=O)Cc2ccno2)C12CCC2 c1(C(N(CCCNC(c2cc(C)sn2)=O)CC)=O)c[nH]c2cc(C)ccc12 Cc1ccc(CNC(C2CCCN(Cc3cnc(O)[nH]3)C2)=O)c(F)c1F CC1=NOC(CNC(=O)CCOCCCNC(C2CCS2(=O)=O)=O)C1 N1(C(C2(OC)CCSC2)=O)CCCC(C2(NC(=O)CCc3cnn[nH]3)CC2)C1 Cc1ccc2[nH]nc(C(=O)NC(C)(CNC(C34CCCC(C3)OC4)=O)CO)c2c1 Cc1noc2nc(C(=O)N(CCCNC(=O)COC(C)C)C)ccc12 c1(-n2c(CC3(F)C(C)C3)nc(C3CCCO3)n2)ccc2ccccc2c1 n1(CC)cc(Br)cc1C(=O)NCCC(C)(C)NC(=O)C=CS(C)=O C1(CN(C)C(C2(Br)CC2)=O)CCCN(C(c2occc2F)=O)C1 CC(C)CC(CNC=O)CC(=O)NC1CC(CNC(C2CCC(=O)C2)=O)C1 N1(C(C(C)OC2CCOC2)=O)CC(=O)NC(=O)C1 c1(OC)cc(C(N2CCC(=CC(=O)Nc3ncco3)CC2)=O)ccc1F C1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)N3)=O)C2)CCC2CCCCN12 CCCCC(C)(F)C(=O)N(CCC(C(C)(C)C)NC(c1c[nH]nc1Br)=O)C c1(OC)ncccc1CC(=O)NC1CCCC(NC(c2ccc(C(N)=O)o2)=O)C1 C1(C)(C(=O)Nc2ccc(OC)cc2)COCCN(C(C)=O)C1.N12CC(C1)C2=O C(=O)(CS(=O)(=O)C1CC1)N1CC(NC(CCN(c2ccccc2)C)=O)C1 Cc1cc(C(N2CCCC2CC(=O)NCC2(O)CSC2)=O)ns1 c1(Cn2cc(CNC(C)(CC(F)(F)F)C(=O)O)nn2)cc(O)n2nccc2n1 c1(C(N2C(C(=O)Nc3c(Cl)ncc(C)c3)CSCC2)=O)cccc2cn(C)nc12 N1(C(C(C(CC)O)(F)F)=O)CCN2CCN(C(c3cncc(F)c3)=O)CC2C1 c1(C(N2CC(C)C(NC(=O)COc3ccn(C)n3)CC2)=O)ccc2nn[nH]c2c1 CC(C)(O)C(C(=O)NCO)NC(=O)C(=O)NC1CCNCCC1(F)F c1(C(=O)NC2CC(NC(C)=O)C23CCC3)cc2cnc(C)nc2nc1O N1(C(C(c2ccccc2)OCC)=O)CCOC(CNC(c2c(Cl)n[nH]c2C)=O)C1 CCC(C)(CNC(=O)COc1ccccc1)C(=O)N(CC(C)C1CC1)C c1(C(N(C2CCCC(NC(c3c(C)snn3)=O)C2)C)=O)cnc2c(c1)CCCO2 c1(C(N2CC(C)C(CNC(=O)C(F)C3CCC3)C2)=O)cc(Cl)c(Cl)cc1O N#CCC(C(=O)N1CCOCC1CNC(C1(C2CCC2)CC1)=O)c1ccccc1 CCC(O)C(C)C(=O)N(CCCCN(C)C(c1ccc(C2CC2)cc1F)=O)C C1(CC(=O)N(CCNC(C2C(C)(CC)C2)=O)C2CC2)CCC(C(=O)NC)CC1 c1(OC)ccc(Br)c(NC(=O)CC2CC(NC(C3CNC(=O)C3)=O)C2)c1 C12(C(=O)NCC(C)(CC(C)C)NC(C(C)=CC3CC3)=O)CCOC1CC(=O)NC2 c1(C(=O)NCC2OCCN(C(C(CC)C#N)=O)C2)cnc(C(F)(F)F)c(F)c1 N1(C(c2c(C)n(C)cc2)=O)CCCC2C(NC(=O)Cc3nncs3)C(C)(C)C12 c1(C(=O)NCCN(C(=O)C=Cc2ccncc2)C2CC2)ccc(O)c([N+](=O)[O-])c1 N1(C(C(C(C)O)(F)F)=O)CC2(COC(CNC(c3ccc(CO)cc3)=O)C2)C1 C(=O)(C1CCCn2ccnc21)NC(C(C)C)CNC(=O)CC1=CCCC1 Cc1nc2c(C(N3CCC(O)(CCNC(=O)C=CC(F)(F)F)C3)=O)cccc2o1 CC(C)CC(O)C(C)C(=O)N1CCC=CC1C(=O)NCC1(O)CSC1 N1(C(C2CC(C)C2)=O)CC2CCCC(CNC(=O)CCS(C)=O)C2C1 c1(C(N(CC)CC)=O)ccccc1CN1CC=CC1.C(=O)(C=CCOCCN(C)C)NC CCC(O)C(C)C(=O)N1CCCCC(C(=O)NC2(C)CSC2)C1 c1(C(N(C(C(=O)N(CCOC)C)C2CC2)C)=O)csc(C)n1 c1(C(=O)NCc2cccc(NC(c3c(C)n(C)nc3)=O)c2)ncnc2c1CCC2 c1(CC(=O)NC2C(CNC(CCS(C)=O)=O)CC2)ccc(Cl)cc1F CC(C(=O)NCC1(C(N2CCC(Cc3cnn[nH]3)CC2)=O)CCCC1)S(C)(=O)=O c1(CC)ccccc1C(=O)NC1CC(CNC(c2ccn(C3CC3(F)F)n2)=O)C1 c1(C(N(C2C(=O)OCC2(C)C)C)=O)cccc(F)c1F.c12cncc(c1)NC2=O N1(C(CC2(N(C(C(CC)C(C)C)=O)C3CC3)CC2)=O)CC(C)(C)CCC1C c1(C(=O)OC)ccc(C(=O)NCC2CC2CNC(c2cc(C)n(C)n2)=O)cc1F c1(C(=O)NCC2(CN(C)C(C3CS(=O)(=O)C3)=O)CC2)cnc(O)c2ncccc12 CC(C)CCC(=O)NC1CCC(C)(CC2(NC(=O)COC3CC3)CC2)C1 C(=O)(C1CCc2ccccc21)NC(CC)(C)CNC(C1CC2(CCCC2)C1)=O c1(OC)cncc(CCC(N2CCC=CC2C(=O)NCC2(C)CCCOC2)=O)c1 Cc1cc(C2CCC2)ncc1C(=O)NC1CCN(C(C2CCOC2=O)=O)CC1F CCC(F)(C(=O)OC)C(=O)N1CC2C(CNC(c3cccc(C)c3)=O)C2C1 C#Cc1cccc(C(N2CCCN(C(C3COCC3(C)C)=O)C(C)C2)=O)c1Cl CC1CCCC(C(=O)NC2CN(C(=O)CSc3ccc(Cl)cc3)C2)CC1 C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CN(C2CCCCC2)C)CC1C n1(CC(=O)NC(C2CCN(C(c3nnc(C)s3)=O)C2)C)ccccc1=O Cc1cc(C)c(C(=O)NC(C2CN(C(c3[nH]cnc3C#N)=O)CCO2)C)s1 c1(C(=O)NCC=CCNC(CCc2cc(C)nc(C)c2)=O)ccc2c(c1)CCCO2 Cc1oc(C(=O)NC2CCN(C(=O)CC(C)(O)c3ccccc3)C2)cc1S(N)(=O)=O N1(C(c2[nH]cc(C(=O)OC)c2)=O)CCCN(C(C2COCCOC2)=O)CC1 C=CCC(C)(CC)C(=O)NCC1(CNC(=O)CC2(C)CCCO2)CC1 CCC(C)C(O)C(C)C(=O)NCC(C)(C)CCC(=O)NCCCc1ccncc1 C(=O)(CC(CC(N)=O)CC(C)C)NC1C(NC(C2(C#C)CC2)=O)CCCC1 N1(CC2(O)CCN(Cc3ccccc3)C2)CCC(F)(F)CC1 N(C(=NCCc1cc(Br)ccc1OC)NCC1(CO)CCCC1)C(CC)C N1(C(C(CC#C)(C)NC(c2cnc(Cl)n2C)=O)=O)CCCC2(CCC2)C1 C1(CCNC(C2CCCC2NC(C2CC2C2CC2)=O)=O)CCCCO1 N1(C(c2cnc(CC)[nH]2)=O)CC2C(CNC(=O)CSC(=N)N)C2C1 C1(CC)CC(C(=O)NC2CC23CCOCC3)CCN1C(=O)CSCCC(C)C c1(-c2ccc(CC)[nH]2)nc(-c2ccc(SC)cc2)nn1CC N1(C(C=COCC)=O)CCCC1(C)CNC(=O)Cn1cc(F)ccc1=O C(=O)(C1=CCC(C)(C)CC1)C(C(C)CNC(=O)N(C)C)=O.C1(N)CCCCC1CC c1(C(=O)NC2(C(=O)OCC)CS(=O)(=O)C2)ccc(O)c(OC(F)F)c1 C1(NC(C(C)SCC)=O)CN(C(c2ccc(OC)cc2Cl)=O)CCC1C.NCC C1(C(=O)NCc2c(C(=O)NC(C)CCC3CC3)cco2)CC2C=CC1O2 N1(C(c2nc(C(C)C)sc2)=O)CCC(OCCNC(=O)C(C)C2CCC2)CC1 CC1CC=C(C(=O)NC2CC(NC(C34CCCC3CCC4)=O)C2)CC1 N1(C(C2(CC)CCN(C(=O)Cn3cnnc3O)C2)=O)CC2CCN(C)C2C1 N1(C(C2(OCC)CCOCC2)=O)CC2CN(C(=O)C=Cc3csc(=N)[nH]3)CCC12 N1(C(C23CCC(OC)(CC2)C3)=O)CC2CN(C(C3CC3(C)C(F)F)=O)CC2C1 c1(C(N(CCN(C(CC(CCC)C)=O)C)C)=O)ccc2c(c1)NCC2 N1(C(c2c(CCC)nco2)=O)CC2CCC1CN2C(C1(OC)CCC(C)C1)=O C1(NC(CC(=C)Br)=O)CC2CC1CN2C(c1c(OC)ncnc1C)=O CCCCC(CCCC)NC(=O)CN(CC(C)C)C(C1CN(C(C)C)C1)=O N1(C(CNC(=O)NCc2ccc(Cl)cc2)=O)CCCC(F)(F)CC1 n1(C(C)C)ccc(=NC(=O)C2C3CCCC3N2C(=O)C(N2CCCCCC2)C)[nH]1 N1(C(C2C(C(=O)Nc3c(C(=O)OC)coc3)C2)=O)CC2CC2C(C(=O)NC2CC2)C1 N1(C(CCNC(C)=O)=O)CCCC(C(C)(O)CNC(=O)COC2CC=CC2)C1 C1(C(=O)NC(c2cncs2)C)CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1C CC1C(NC(=O)CCCC(F)(F)F)CC2CCC1N2C(c1cncc(Cl)c1Cl)=O C(=O)(C(CC(C)C)ONC(c1cn(C)c(=O)cn1)=O)NCCc1c(C)nccn1 Cc1cn2ccc(C(=O)N(C3CN(C(C4(C)CC(O)CN4C)=O)C3)C)cc2n1 c1(C(=O)NCC2(NC(CC3ON=C(CC)C3)=O)CCOC2)cccc2nncn12 C1(C(F)(F)F)(C(=O)NC(C)CN(C(C2CN(c3nncs3)C2)=O)CC)CCCS1 C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)C=Cc2cnn(C)c2)CC2(CC2)C1 c1(NC(=O)NC)ccc(Cl)c(C(=O)NC2C(CNc3ncnc(NC)c3F)C2)c1 C1(C(=O)NCC(=O)Nc2c(F)cccc2F)CCc2ccccc2C1 c1(CC(=O)NCC(O)CNC(c2cc(F)c[nH]2)=O)ccc2c(c1)OCCCO2 Cc1cc(NCc2ccc(Br)cc2)nc(N2CCCC(c3nc(C)c(C)[nH]3)C2)n1 C1(NC(C(C)C)=O)CCN(C(=O)C(O)CC2CCOCC2)C12CC2 c1(C(N2CCC3CN(C(C=CCC)=O)CC3C2)=O)cc(Cl)cc2ccncc12 c1(OCC(CNC(c2cccc(OCC)c2)=O)O)cnc2ccccc2c1 c1(C(=O)NCC2CCCC(NC(c3nccc(OC)c3)=O)C2)cc(C)n(C)c1C c1(OC)cc(C)nc(N2CCC(C)C(NC(=O)C=Cc3cncnc3O)C2)n1 CC1CCCC(CC(N2CC(CNC(=O)CCCCNC(N)=O)CC2C)=O)C1 c1(N2CCC(N(CCC3CCCOCC3)C)C2)cc(Nc2ccccc2)nc(C)n1 CC(CCC(C)(C)C)C(=O)N1CSCC1C(=O)NC1CC12CCCC2 N1(C(c2ccc(N)c(Cl)n2)=O)CCC2CC2(NC(c2csc3nnsc23)=O)CC1 C1(N(C(C(CC)C)=O)C)CN(C(=O)CC2CCCCC2)CCC1C C1(NC(C(C)NC(c2cccs2)=O)=O)CCN(C(=O)C(C)C2CC2)CCC1(F)F Cn1nccc1CCC(N1CCC1(C)C(N1CC(C(=O)NC2CC2)C1)=O)=O N1(CC(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)CCC(=O)NC1=O N1(CC=C)CCC2(CN(C(c3cccc(C)c3F)=O)CC(C)O2)C1 c1(C(c2n(CC)nnn2)NCCC(C)COC)ccc(F)cc1 N1(C(CCCOC)=O)CCCC1(C)C(C)(C)C(=O)NCC1(C(C)C)CC1 Cc1cc(=O)c(C(=O)NC(C)(CNC(=O)CCOCC(F)F)CC(C)C)cn1C C1(C(=O)NCC2N(C(C3(O)C(C)(C)C3)=O)CC2)CC12CCCCC2 c1(C(=O)NCC(F)F)ncn2ccccc12.c12ccc(cc1)[nH]2 C1(NC(=O)CNC(=O)C2CC2)CC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC12 c1(NC(C2N(C(c3c(C)nccc3)=O)CC2)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(c2cc(C)oc2C)=O)CCCC(F)(CNC(C2(C)CCCOC2)=O)C1 C(=O)(C(C)(C)C(F)F)NC1C(CNC(c2c(C)n(CC(F)F)nc2)=O)CCCC1 Cc1ccc(C(=O)NCCC2CCC(NC(=O)C3=COCCC3)C2)c(C)c1 C1(N(C(=O)CCN2CCC(F)C2)CC)CCN(C(C2COCCOC2)=O)CC1 N1(C(C2N(C(c3cc(C(C)=O)[nH]n3)=O)CC(F)C2)=O)CCOCC(F)(F)C1 c1(-c2n(CCN(C)C)nc(-c3cc(F)cc(F)c3)n2)n[nH]c2c1COCC2 c1(CN2CC(c3ccccc3)(NC(CSCC)=O)C(C)C2)ccc2sccc2c1 c1(OC(C)C)ccc(Cl)c(-c2ccc(CN3CC4CCCCC4C3)c(F)c2)c1F O=S(=O)(c1ccc(Br)cc1F)NC1CCC(Nc2ncnc3sccc23)C1 c1(C(=O)NCC(CCCC)NC(C2CCC(N=[N+]=[N-])C2)=O)cc(F)cc(F)c1O CC1(C)CCCCC(C(=O)NCCCC2CC2(F)F)C1 C1(NC(=O)C(CC(F)F)C2CCC2)CCCCCN(C(c2ccoc2Cl)=O)C1 CC(C)CCCC(C)C(=O)NCCCCC(CO)NC(=O)COC(C)(C)C C1(NC(c2noc(CC)c2C)=O)CC2CN(C(=O)C3=NOC(C)(C)C3)CC2C1 N1(C(c2c(C)noc2)=O)CC2CCN(C(C3CCC(C)(C)CO3)=O)C2C1 C1(CC)CN(C(=O)C(C)(C)CNC(C)=O)CCN1C(C1C2CCC1CC2)=O N1(C(C(C)OCCCCCC)=O)CCC(NC(C2(COC)CCCC2)=O)C(F)C1 C=CCC(CNC(C1CCCN1C1CC1)=O)NC(=O)CSc1nnc(S)s1 C1(C(N2CC(NC(C3(c4c(OC)ccc(Cl)c4)CC3)=O)C2)=O)CCC2(CCC2)OC1 c1(CC(=O)NC2C(C)N(C(=O)C(C)O)CCC2)cc(F)c(F)cc1F c1(NC(C2CCC(Nc3ncc(OC)cn3)C2)=O)cc(C)cc(Cl)c1 CCC(C)C(C)C(=O)NCC(C)(C)NC(c1ccc(N2CCC(C)CC2)nc1)=O N1(C(c2ccnc(C)c2N)=O)CC2CCC1CC2NC(=O)CC1COCC(C)O1 N1(C(C(C)N2CCCC2)=O)CCCCC1c1ncon1.N1(c2nncs2)CCCC2(CC2)C1 c1(C(=O)NC(C2CCN(C(C(CC)SC)=O)CC2)C)cc(N)cc(O)c1C c1(OC)cc(O)c(C(=O)NC2CN(C(=O)C(C)NC(N)=O)CC2C)cc1OC C1(C(=O)NC(c2nccs2)CC)CC(C)(C)CCN1C(c1ccc(CO)o1)=O n1(CC)cccc1C(=O)NCCC(C)NC(c1ccncn1)=O N1(C(CC(c2c(C)cccc2)C)=O)CC(NC(=O)C=CC(=O)N(C)C)CC(F)(F)C1 N1(C(C(Cc2ccco2)OC)=O)CC2CCCC2(NC(C2CC2(F)Cl)=O)C1 CC(C)(CC(=O)N1CCCC(NC(=O)CCn2cc[nH]c(=O)c2=O)C1)C(F)(F)F C(C(=O)NCC1CC1C=C)(C(C)(C)O)NC(C=CC(CC)C)=O C1(C(=O)NCCCO)CCC(C)C1.C1(CC)(C(=O)N(CCCO)CCO)CCC1 C=CCC(CNC(c1cnoc1-c1ccccc1)=O)NC(C1(C)CC1)=O Cc1ccc2[nH]c3c(c2c1)CN(C(C1CN(C2CCCCC2)CCC1O)=O)CC3 C1(CCC=C)CCCC1N=c1[nH]c(N2Cc3ccccc3C2)nc2ncn(CC)c12 c1(SC)cc(C(N2CC(C(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)c(C)o1 C12(C(=O)NC(CC)CNC(=O)Cc3nc(=N)[nH][nH]3)CC(CC(C)O1)C2 CC1CC(C(=O)N(C2CCN(C(=O)CSC(=N)N)CC2)CC2CC2)CCO1 N1(C(C(CCSC)O)=O)CCC(CC(F)F)(CO)CC1 N1(C(CCCCCN(C)C)=O)CCC2(CC1)CC2C(=O)NCC1(C)CCCOC1 C(=O)(C(F)(F)C(O)CCCC)NCC(CCCC)NC(=O)CCCSC(C)(C)C CC1(C)CN(C(=O)CCc2ccoc2)CC1CNC(=O)CSC(F)F N1(C(C(C)CN(C)C)=O)CCCC2CN(C(C3SCCS3)=O)CC12 c1(NC(CC2OCCN(Cc3cccc(OCC)n3)C2)=O)c(C)cc(O)cc1O N1(C(C2C(C#C)C2)=O)CC(CNC(=O)CN(CC(=O)NC)C)OC2(CCC2)C1 CN1C2CCCC1CN(C(C1CC1C1CN(C(c3c(C4CC4)noc3C)=O)C1)=O)C2 c1(NC(N(C2CCN(C)CC2)Cc2ccc(C#N)cn2)=O)cn2ccc(Cl)cc2n1 C(=O)(CC(C(F)(F)F)SC)NCC1(CC)CCCCO1.C12(CCC1)C(=O)N2 C(CCNC(C1CC1(C)Br)=O)(C(C)C)NC(C(CC)n1nccc1C)=O C1(C(N2CC(C)OCCC2)=O)CC2CCCC2N1C(=O)CCc1nncs1 c1(C(=O)NC(CC(=O)OCC)Cc2cccc(F)c2)cccc([N+](=O)[O-])c1Cl c1(CNC2(CNC(C3(CC)CCC3)=O)CC2)ccc(OC)c(Br)c1 c1(-n2cc(CNC(C3C(C(=O)OC)C3)=O)nn2)cc(F)cc(F)c1 c1(OC)c(Cl)nc[nH]c1=NCC12CCCCC1CN(C(=O)CC1(CO)CC1)C2 C(CN=c1ccc(-c2cccc(OC)n2)c[nH]1)Nc1cc(OCOC)ncc1 N1(C(C2(CN(C)C)CC2)=O)CCCC2(CCCN2C(C2(C3CCCO3)CC2)=O)C1 Cc1ccc(-c2cn(CC3CN(C(c4ccc(C)cc4C)=O)C3)nn2)c(C)c1 C1(CC)C(C(=O)NCC2CCC2(F)F)CCCN1C(=O)CCC1CC1(F)F c1(C(N2CC(CNC(CC(C)OC)=O)C3(C2)CC3)=O)cc2ccccc2o1 Cc1nc(CCC(=O)NC(C2CN(C(C3(C)CC3(F)F)=O)C2)C)oc1C c1(CCC)ncoc1C(=O)N(CCCNC(C1CCCS1)=O)CC1CCCC1 Nc1cc(F)cc(Cl)c1C(=O)NC1CCC2CCN(C(=O)CC3CCCCC3)C12 N1(Cc2cc(C)[nH]n2)C(C(N2CCC(Nc3ncccn3)C2)=O)CC2CC12 C(=O)(C(C)CC(C)(C)C)N(CCNC(c1c(C)n(C)cc1)=O)CCOCCO C1(CCNC(CCC=C)=O)CN(C(C)C(=O)NC2CC2)CCS1(=O)=O C1(CN(C(C(C)OC)=O)C)CCN(C(C2CC2C(F)(F)F)=O)CC1 n1(CC)cc(NC(=O)CC2CCCN(C(=O)C(=O)c3ccco3)C2)c(C(N)=O)n1 C1(C)(C(N2CCC(O)(CNC(c3cncc(CC)c3)=O)C2)=O)COCC1(F)F C(=O)(C(C)Cc1cnco1)NC(c1cn(CC(=O)OC)nn1)C1CC1 C=CC(CC(=O)NC(C)CNC(C1(Cc2cnn(C)c2)CC1)=O)c1ccccc1 CC(C(=O)N1CCN(CC2(NC(c3cncc(C(N)=O)c3)=O)CC2)CC1)C(C)O CCC(C)CC(C)C(=O)N(C1CCN(C(C2CC23CCCC3)=O)CC1)CC1CC1 Cc1cn2c(n1)C(C(=O)NC1CC(CNC(c3ccc(C)c(N)c3)=O)C1)CCC2 Cc1cc2[nH]c(C(N3CC4(C3)CN(C(C3CCC3c3nc(S)n[nH]3)=O)C4)=O)cc2s1 C=CC(C)(CC)C(=O)N1CC2C(CNC(=O)CCCF)C2C1 c1(NCCc2cccc(C(=O)O)c2)c(Cl)cccc1[N+](=O)[O-] c1(C(N2CCC(O)(CNC(C34CCC(C3)C4)=O)C2)=O)ccc(Cl)cc1Cl C#Cc1c[nH]nc1C(=O)NCC1CC(NC(=O)C(C)CC=C)C1 c1(C(N(CC(=O)NCCN(C)CC)CC(C)C)=O)cc[nH]c2nccc1-2 c1(C(N2CCCC(NC(c3cc(CC)n(C)n3)=O)C2C)=O)ccnc2c1CCC2 Cn1cc(C(N2CC(CNC(=O)C(=O)NCC3CC3)C(F)(F)C2)=O)c(O)nc1=O C1(CNC(C(CC)O)=O)(NC(c2ccc(C(N)=O)nc2)=O)CCOCC1 C1(OC)CC(CNC(=O)Cc2cscn2)N(C(c2cccc[n+]2[O-])=O)C1 N1(C(c2cnc(COC)[nH]2)=O)CC2(CCCC(CNC(=O)CC=C(C)C)O2)C1 N1(C(C(C(C)C)C(C)NC(=O)C=CCN2CCCC2)=O)CCC2CCC(C1)N2C c1(-c2cn(C(C)C(=O)NC(C)CCCCCC3CC3)nn2)c(F)cncc1F C1(NC(c2nccc(C)c2)=O)CC2CC(C1)N(C(=O)COc1ccsn1)C2 N1(C(c2c(C)ccc(F)c2)=O)CCC2CC2(C(N2CC(N3CCCCC3)C2)=O)CC1 N1(C(C2(CC)CCCN2C(c2cn3ccccc3n2)=O)=O)CCCCCCC1C N1(Cc2cn(CC(OCC)OCC)nn2)CCC(C)(NC(=O)NC2CCO2)CC1 CCCCCC(C1CC1)NC(=O)C(CC1CC1)NC(c1nocc1Cl)=O C(=O)(CCCCC(=O)NCCC1CCCN1C(=O)CN(C1CCCC1)C)NC C(=O)(C1(C)COc2ccccc21)N1CCCCC(CNC(C(C)(C)CO)=O)C1 CCC(C)C(O)CC(=O)N(CCC(=O)Nc1cnc2[nH]cnc2c1)CCCO C=Cc1cnn(C)c1C(=O)NC1CC1CNC(c1cnc(C)nc1C(C)C)=O C1(CNC(C2(CCC=C)CC2)=O)CCN(C(c2ccc(CC)nc2C)=O)C12CC2 c1(C(N2CCC(CCNC(CCc3onc(CC)n3)=O)C2)=O)cnc(O)cc1C C12(NC(c3cccnn3)=O)CCCC1N(C(c1cncc(O)c1)=O)CC2 N1(C(c2c(C)ocn2)=O)CCN(C(CNC(C2CCCCN2C)=O)C(F)F)CC1 c1(OC)ccc(CN2CC3C(C2)N3C(c2cc(C(F)(F)F)c[nH]2)=O)cc1 C(C)(CCN(C(=O)C(C)SCC(C)C)C)NC(CN(CCC)C)=O C1(NC(C(c2ccc(C(F)(F)F)s2)N(C(C)COC(C)C)CC)=O)CC(F)(F)C1 N1(C(C(CC)C(C)C)=O)CC2CN(C(C3CC3c3cccs3)=O)CC(C1)O2 C1(NC(C2C(C)CN(C(=O)CNC(N3CC=CC3)=O)C2)=O)CCC(C2CC2)C1 C(=O)(C(O)CCC(C)C)NC1CN(C(C2(OC)CCSC2)=O)CC1F N1(C(c2n(C=C)nnc2)=O)CC2C=CC1C(C(N1CC3CCCC13)=O)C2 N1(C(c2sc(C)c(-c3ccc(F)cc3)n2)=O)CC(N)CCc2ccccc21 c1(C(CNC(c2ccc(Br)cc2)C)NCC(=O)NC(CC)CO)ccc(Cl)cc1Cl O=C1CCC2(CC1)CCN(CCC1CC3(CC3)C1)C2 c1(SCc2ccnc(C(CC)C#N)n2)cccc(P(C)(C)=O)c1 c1(CC(=O)NC23CC(NC(C4COCC(C)O4)=O)(C2)C3)ccc2c(c1)COC2 c1(C(=O)NCC2N(C(c3cc(C(C)(F)F)on3)=O)CC2)ccccc1F N1(C(=O)NCC)CC(C(=O)NCCCN(C(=O)CN)C)C1 C1(C)(C(=O)NCC(CC)NC(c2cn(CCOC)nc2)=O)CC(OC)(OC)C1.CC CCC(CCC(=O)N1CC(c2ccccc2)(NC(C2C=CCC2)=O)C1)OC c1(OC)ncc(C(N2CCC(N(C)C(c3cn(C)nc3SC)=O)C2)=O)cc1Cl N1(C(CNC(C)=O)=O)CCCCC1C1CCCN(C(C2(C)CC2)=O)C1.C1(=O)CCN1 CCC(C)CC(=O)NCC1COCCC1NC(C1(Nc2ccccc2F)CC1)=O CCC(CC)C(C)C(=O)N(C1CCCN(C(C2(O)CCC2)=O)C1)CC C(CC(C(=O)NC(C1CC(F)(F)C1)C)NC(c1cccnc1S)=O)SC CC1(C)C(=O)NC2CCCN(CC(c3cn(C4C(F)C5CCCOC45)nn3)N)C12 C1(COC)(CNC(C2CCSCC2)=O)CCN(C(C2COCCO2)=O)C1 C1(NC(COCCC)=O)COCCC1C(=O)N(CCCO)C(C)C c1(COC)ccc(C(=O)NC2(CCCNC(=O)C(n3ccc(C)n3)C)CC2)s1 C(=O)(C1COc2ccc(Cl)cc21)NCC1CC2CN(c3nccc(C#N)n3)CC21 C12CCCN(C1)C2.c1(NC(C2C(C(=O)O)(CC)C2)=O)ncoc1C(C)(C)C c1(C(N2CCC(C(C(=O)NCc3cccc(F)c3O)F)C2)=O)cc(O)ncc1F C1(C(=O)NCCOC(=N)O)CN(C(C2CCCC2C2CC2)=O)CC1(F)F CC1(C)OC2(C(=O)NC3CC3NC(C3(C4CCCCO4)CCC3)=O)CCC1CC2 CCC(C)CCCCC(=O)NCCC1CCCN(C(c2cnc(COC)s2)=O)C1 c1(C(=O)NC2C(SC)CN(C(C3(C(N)=O)CCC3)=O)C2)nccc2cccnc12 C(CC(C)C)(C(=O)NC(c1csnn1)C)ONC(C(C1CCOC1)OCC)=O c1(C(=O)NCC(C)CN(C)C(C2CC2C(N)=O)=O)cncn1C C1(NC(=O)CCc2ncc[nH]2)CCCC12CN(C(C13CCCC1CCC3)=O)C2 C1(C(N(CCOCCCNC(CC=CCCCCC)=O)C)=O)CCNC(=O)C1 O=C(N=c1[nH][nH]c2ccc(F)cc12)c1cc(F)c(F)cc1.C(F)(F)C(F)(F)Cl N1(C(c2c(C)sc(-c3nc[nH]n3)n2)=O)CC=C(C(=O)N2CC(C(N)=O)C2)CC1 N1(C(=O)Cn2cnc(Br)n2)CCCN(C(=O)C=Cc2ccco2)C(CO)C1 Cc1ncnc(C)c1OCC(=O)NCC(C)(C)NC(c1ccsc1C#N)=O C(CC(C)C(=O)N(CCCNC(C1CC(OC)C1)=O)C)=CC c1(C(N(C2CCN(C(c3ccc(CN(C)C)[nH]3)=O)CC2)CC)=O)cc(=O)cc[nH]1 c1(C(=O)NC(c2ccccc2)C(C)NC(C=C=C(C)C)=O)cnc(C)c(C)c1 C12(C(=O)NC3CCN(CCCNC(C4CC(O)C4)=O)CC3)CCCC1CCC2 C1(C(=O)NCC(Cn2cc(-c3cncn3C)nn2)OC)CC(C)N(C)C1 C(=O)(CCC(C)(C)C)NC1C2CN(C(c3c(CC)nccc3)=O)CC21 N1(C(CN(C(C)C)C)=O)CCN(C2CN(C(=O)CC(O)C3CCCC3)C2)CC1 c1(N(CCOC)C)nc2c(c(=NC3CCN(c4cccc(Cl)c4)C3)[nH]1)SCC2 N1(C(CCC=C(C)C)=O)CCC2(CC1)CC(NC(=O)CC1CCC(C)CC1)C2 N1(C(c2c(C(F)(F)F)nc(C)o2)=O)CCC2(CC2NC(C2C(C)C2(F)F)=O)C1 CC(C)(O)C(F)(F)C(=O)N1CC2(CCNC(=O)COC3CCC3)CCC1CC2 C1(CNC(C=C(C)Cl)=O)COCC2(CCN(C(c3ncn(C(C)C)n3)=O)C2)O1 c1(-n2c(CCCc3ccc(CC)cc3)nc(C(CCC)C)n2)cc(F)cc(F)c1 c1(C(=O)NCC(CN(C(C(c2ccccc2Cl)OC)=O)C)C)ccc(C)cc1Cl Cc1ccc(C)c(C(=O)NC(C)(C)C=CC(=O)NC2CCN(C)CC2C)n1 Cc1ccccc1C(C)(C)C(=O)N(C1CCC(CNC(=O)CC(C)O)CC1)C c1(C(=O)NC(=O)CCSC)ccc(C)cc1.CCC1C(=O)N2CC(O)(C2)CN1C C(=O)(C(C)(CC)CCC)NC1CC(C(N(C(CC)C)CC)=O)C1(C)C N1(C(COCCC#C)=O)CCC2CN(C(=O)C(CC)n3ccnc3)CC2C1 N1(c2n(CC(=C)C)c(C3CCCN3CC(F)(F)F)nn2)CCC(C)OC1 N1(C(C(COC)C)=O)CCCCC1CNC(=O)CCNC(c1c(O)noc1C)=O C12CCCC1C(=O)NC2.CC(C(F)F)=CC(=O)NCC1CCC1 CC1(C)C(NCc2nsnc2O)CC1CC(=O)NC1(CO)CCCCC1 CC1(C)CC2(CC(C(=O)NCc3cccc(CNC(C4CC4(F)Cl)=O)c3)C2)C1 C#CCC(CC(=O)NCC12CCCCC1C2)NC(c1c[nH]nc1[N+](=O)[O-])=O C12(CC3(CC3)C1)C(=O)NC2.c1(C=O)cc(C)n(C)n1.N1(OCC)CCC(C)C1 O=S(=O)(c1ccc(NC2CCCC3(C2)OCCO3)c(F)c1)NCCC1CCCC1 c1(C(=O)NC(CNC(CCC=CCC=C)=O)CC(C)C)cc(C)ccc1O N1(C(C(C)CN(C)C)=O)CC2CN(C(c3cc(C(F)F)ccc3Cl)=O)CC2C1 C1(C(=O)NCC2N(C(CC(CC)CC)=O)CC3(CC3)C2)CCc2c(nnn2C)C1 N1(C(C(C)NC(=O)CC(C)(O)C(F)(F)F)=O)CCC12CCC(O)CC2 N1(C(CC2(CS(N)(=O)=O)CC2)=O)CCC(F)(C(=O)NCCCO)CC1 C1(NCC(CC)C2CCOCC2)CCN(C(C2(C(F)(F)F)CC(O)C2)=O)CC1 n1(CC(N2CC3CCC3(C(N3CCC(F)(F)C3)=O)C2)=O)nc2ccccn2c1=O C1(CNC(C(C)OCC#C)=O)CCCC1NC(C1(CNC(C)=O)CCC1)=O c1(C(N(CCN(C(c2ccc(Cl)s2)=O)CC)CC)=O)cnc(O)c(OC)c1 C1(n2ncc(NC(CC(O)OC(C(C)Cc3ccnn3C)=O)=O)c2)CCN(C)C1=O c1(OCC(C2CCC(O)CC2)(OCC)OC)ncnc2[nH]c3ccccc3c12 Cc1cnc(CCC(n2cc(-c3n(CC(=O)OC)nc(C4CC4)c3)nn2)C)cn1 Cc1nc(CNC(=O)C(C)N(C(=O)C(CO)N(C)C)CC2CC2)c(C)s1 CC1CC(NC(=O)CCC(N)=O)CN1C(=O)CCCc1ccsc1 c1(NC(C2(C)CCN2C(C2CC2c2ccccc2)=O)=O)cnn2ccccc12 CC(C)C(O)C(=O)NCCOC(CNC(=O)C(C)Oc1ccccc1)(C)C N1(C(CCc2cc(C)no2)=O)CCC2(CCCN(C(=O)COC(F)(F)F)C2)C1 C1(NC(C=CCCC)=O)CCS(=O)(=O)C12CN(C(c1c[nH]nc1F)=O)C2 c1(CC)ccc(NC(C2OCCC2CNC(=O)C(C)OC)=O)c(F)c1 CC1CCC=CC1C(=O)NCC(C1COCCN1C(=O)C(O)C1CC1)(C)C C1(CCNC(c2n(CC#C)ccc2)=O)CC(OC)CN1C(c1cncc(N)c1)=O CC(CC1CC1)C(=O)N1CC(C(C)O)(CNCCNC(=O)C=CC(C)(C)C)C1 C(=O)(C1CCc2cccc(=O)n21)Nc1ccc(NC(=O)OC(C)(C)C)cc1 N1(C(C(C=C)(C)C)=O)CCC2CN(C(c3n[nH]cc3C(C)C)=O)CC2C1 N1(C(CCN(CC)CC)=O)CC(CC(=O)NCc2ncccn2)CC1C c1(CC2(CC(=O)NC(C3CCN(CC)C3)C)CC2)cccc(C(F)(F)F)c1.C(N)=O c1(C(=O)NC2CN(C(c3ccc(C#C)cc3)=O)CC(C)C2)cc(F)cc(F)c1O C(C(=O)N=c1ccn(C(C)(C)C)[nH]1)(C1CCC1)NC(C(C)=CCC)=O S(=O)(=O)(c1ccccc1-c1cncnc1)N1CC(C(=O)OC)C2(C1)CCC2 C1(C(N(C)C)=O)CC(F)(CNc2cc(-c3ccccc3)co2)C1 C=CC(C)(O)CC(=O)NCC1CC2(C1)CN(C(c1ccc(C(C)C)o1)=O)C2 N1(C(COC)=O)CCOC(C2CN(C(=O)CCC(N)=O)C2)C1.C12(CC1)CCCO2 C(=O)(CCCC(=O)NC1CC(F)(CNC(c2csnc2Cl)=O)C1)N(CC)CC CC1(C)OC2CN(c3ncnc(N4CC(CCO)OC(C)(C)C4)c3C)CC2O1 C(=O)(C(C)(C)CCF)N1CC(C(N(C)Cc2c(C)n(C)nc2)=O)C(F)C1 C1(C(=O)NC(CNC(CC=C)=O)CC)CC(F)CN1C C1(CNC(CCC(C)O)=O)CN(C(=O)C(CO)c2ccccc2)CC1(C)C c1(C(=O)NCC(C(=O)NC)C)c(CNC(=O)CC2CCSCC2)nnn1C c1(CC)onc(C)c1C(N1CCC(OCCCNC(C2CC2C(C)O)=O)CC1)=O C(=O)(CCCN(C)C(C)C)N1C(CC(=O)N(CC(N)=O)CC)CC1 CC1(F)CN(C(=O)C=CC2CCOCC2)CCN(C(c2cccc(Br)c2)=O)C1 C1(C)(CC)C=C(C(=O)N(C2CN(C(c3cnn4cc[nH]c34)=O)C2)C)C1 CCC(CC(C)C)C(=O)NC1CCN(CCCNC(c2csc(C)c2C)=O)C1 c1(OC)ccc2c(c1)N(C(c1cccc(OC3CCC(=O)N3)n1)=O)CC(=O)N2 CN1CC=C(CC(=O)N2CCC(C)(C)C2C(=O)NCCN2CC=CCC2)CC1 c1(OC)cc(OCN)c(CN)cc1F.C12(CCC1)C(=O)NC2.C(C(C)C)OC c1(CC(=O)NC2C(OC)CN(C(C3CC34CC(O)C4)=O)C2)ccc([N+](=O)[O-])cc1 C1(C)(C(=O)OCC(=O)Nc2nnc(CC(C)C)s2)CCC2(CC1)CC2 Cc1cc(CNC(=O)C=Cc2cn(C)nn2)oc1C(=O)NCCN(C)C C1(NC(CCC(C)=O)=O)COC2(CCN(C(=O)Cc3cccc(O)c3)CC2)C1 c1(C(N2CCC(CCNC(=O)Cc3ccns3)CC2)=O)n[nH]c2c1CCC2 C1(NC(C2(OC)CCC(C)C2)=O)CN(C(C2(C)CSC2)=O)CCC1C C1(CCN(CCC)CC)CCN(C(c2sncc2C)=O)CC1 C(=O)(C(C)S(C)(=O)=O)NCCCN(C(CCSCC)=O)C1CC1 C12(C(=O)NCC(C(N3CC=C(C)CC3)=O)CC3CC3)CCCN(CC1)C2 C12(CC(=O)NCC3(CSCC)CC3)CCC1CN(C(=O)C(O)CC1CCCC1)C2 C1(CC(=O)NC)CN(C(C2(C(C)C)CC2)=O)CCN1C(N)=O.c1(C(=O)N)[nH]nnc1C C12(C(=O)NCC3(C(N4CCN(CC)CC4)=O)CC(=C)C3)CCCC1C2(F)F C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)C(N2CCOCC2)C)CCC1(F)F C12(CNC(C3N(C(CCC)=O)CSC3)=O)CC(NC(=O)C=CC3CC3)(CCO1)C2 c1(CC(=O)NCC(CC)NC(C2CC(N(C)C)C2)=O)ccnc(Cl)c1F C12(C(=O)NCc3cn(CC)nn3)C(NC(=O)CC3CCSCC3)C3CC1C2C3 c1(C(N2CCC(CC)C2CNC(=O)C2=CCCC2)=O)cc(C)nc(C)n1 C1(C(N2CCCCC(Cc3cccc(F)c3)C2)=O)CCC2(CN(CCO)C2)O1 C(=O)(CC(C(F)(F)F)NC(C1(C)CNC(=O)N1)=O)NCCC(C)N(C)C c1(C(=O)NCC2C3CN(C(=O)CCc4cscn4)CC23)c(O)ccc(Cl)c1F CCCCCCCC(=O)N1CCC(C(N2CCC(NC(C)=O)C2)=O)(CF)C1 C#Cc1ccc(C(=O)NCC2CCC(NC(c3cnnn3C(C)C)=O)C2)cn1 N#CC1OC2(Cc3cn(C(=O)Nc4cccc(-n5ccnc5)c4)nn3)CC1C2 C(CCCCC(=O)NC1(C(=O)N(C)C2CC2)CCCC1C)NC(C)=O CCCC(C(=O)N1CCCC1=O)C(C)C N1(C(=O)NC2CCCN(c3ccc(Cl)nn3)C2)CCC(O)C12CCC2 N1(C(c2cc(OC)c(F)cc2)=O)CC2CCC(NC(c3cc(Cl)sc3Cl)=O)(C2)C1 N1(C(CC(C)n2cccn2)=O)CCCC2CCN(CCc3ccccc3)CC12 C(=O)(CCCCN(C)C(C1(CCN(C)C)CC1)=O)NC(c1nn(C)c(=O)o1)C c1(C(=O)NCC2CC(NC(C(=O)NCC)=O)C2)ccc(Br)c(C)n1 c12cn(C)nc1C(=O)NC2.C(CC)(C(=O)OC)N(C(C(C)NC(C=C)=O)=O)CC c1(C(N2C(CCCNC(CCC#C)=O)CCCC2)=O)n[nH]c2ccc(OC)cc12 CC(C)(CNC(c1cc(CCNC(c2c[nH]nc2Cl)=O)on1)=O)CO c1(NC(=O)NC(C)C(c2ccccc2)O)cccc(Br)c1.N12CCC(C1)CC2=O CC1CCc2ccccc2N(Cc2ccc(C#N)cc2)C1 c1(C2(C(N(CCN(C(c3cncc(NC)c3)=O)C)C)=O)CC2)ccc(F)cc1C N1(C(C2(C)CCCC2)=O)CCCC2(CCC(NC(=O)C=CC3CCCCC3)C2)C1 N1(C(c2cc(C)c(C)[nH]2)=O)CCCCCC1CNC(C12CC=CC(C1)OC2)=O C1(C(=O)NCC(C(C)C)(C)NC(=O)C2=NNC(=O)C2)CCC(S(N)(=O)=O)CC1 c1(C(=O)NCCCN(CCCNC(C2CC2Cl)=O)C)ccnc(OC(F)(F)F)c1 C1(C(=O)NCCN(C(=O)C(F)(F)C(O)C(C)C)CC)CCCCC(C)(C)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2(C1)CN(C(=O)CCc1cnc(O)[nH]1)C2 c1(C(N2CCCC(N(c3c(C)cnc(C)n3)C)C2)=O)ccc2cncn2c1C c1(C(=O)NC2(C)CC(NC(C(c3cccc(C)c3)O)=O)C2)ccc(F)c(Cl)c1 C12(CC(=O)NCC3C(NC(C4(C)CCCC4)=O)CC3)CC3CC(C1)CC(F)(C3)C2 c1(-c2cccc(OCC=CC)c2)ccc2cc(Nc3[nH]cnc3CC)ncc2c1 c1(OC)ccc(F)c2[nH]c(C(N3CC4(CC4)CC3CCN)=O)cc12 c1(OC)ncc(C(=O)NC2CCCCC2CNC(=O)C=Cc2ccccn2)cn1 Cc1ncc(C(=O)NC2CN(C(=O)CCCn3ccnc3)CC2C)cn1 N1(C(CSC(=N)N)=O)CCN(C2CN(C(=O)CCC3CC3)C2)CC1 C=CCCCCCC(=O)NC12CCC(C1)N(C(C1CCN(C)C1=O)=O)C2 c1(C(=O)N(CCC(N2CCCCCCC2)=O)C2CC2)c[nH]c2ccccc12 c1(C(=O)NCC2(NC(=O)C(=O)Nc3ncc[nH]3)CCOC2)[nH]nc2ncccc12 CC(C)C(C(=O)NCC1CC(O)C1)C(C)NC(=O)C(C)C1(O)CCC1 c1(C(=O)NC2(C)CCN(C(=O)Cn3cccn3)C2)cc(=N)[nH]c(Cl)n1 O=C1NC(=O)C(CCC(N2CC(O)(CCNC(=O)Cc3ccco3)C2)=O)N1 Cc1noc(Cl)c1CC(=O)NCC1CC(CNC(=O)CNS(=O)(=O)N(C)C)C1 c1(CC)nc2cc(F)ccc2cc1C(=O)NC1CCCN(C(C2SCCCS2)=O)C1 C1(NC(c2c(CCC)occ2)=O)CCN(C(=O)C(F)OC(F)(F)F)C12CCC2 C=CC(C)C(=O)NC1CCN(C(C2CCC2C#N)=O)C1 C1(NC(c2nc(Br)c[nH]2)=O)C2CCN(C(C3C4CCCCC34)=O)CC12 c1(C(=O)NC2C(CNC(C3CCC(OC)CC3)=O)C2)ccc(Br)cc1N C1(C(N2CCCC(C3(C)COC(=O)N3)C2)=O)CN2CCC1(F)CC2 C12(NC(CCNC(=O)OCC)=O)CCCC1CN(C(c1ccc(C)c(F)c1)=O)C2 CC1CC(=O)NCC1C(=O)N(CCCCN(C)C(C1(C2CC2)CCC1)=O)C C1(C(N(C(=O)CC2CCCC2)CCNC(=O)CS)=O)CCC2(CCOCC2)O1.CC N#Cc1ccc(CC(=O)NC2CC2NC(C2(O)CCCCC2)=O)s1 c1(CNC(c2c(C)oc(Cl)n2)=O)cnc2c(c1)CNC2=O N1(C(c2cc(C#C)c(C)cc2)=O)CCC2(CCN(C(C3(C(C)C)COC3)=O)C2)C1 N1(C(C(CSC)C)=O)CCC(C)(C)C1C(=O)NCC1(CCO)CC1 C1(F)(CNC(c2nc(C)[nH]n2)=O)CCCN(C(C2CCN(C3CCOC3)C2)=O)C1 N1(C(Cc2nc(C(C)C)sc2)=O)CC2CC1CN(C(C13CC4CC1C3C4O)=O)C2 N1(C(c2cc(Br)cc(C)c2C)=O)CCC2CCN(C(=O)CC3CCCO3)CC12 C(=O)(CC(C)(C)NC(=O)COCC(C)C)N(C1(C)CCCO1)CC CCC(CCC(=O)NCC1OCCC1C)NC(=O)CN(C(=O)C(C)C)C c1(SC(c2ccccc2C)c2ccc(CNC)o2)c(C)cc(C)cc1C C(C)(CCC(=O)NCC1CCN(C(=O)CC2CCOCC2)C1)OC N1(C(C23CC(C(=O)OC)(C2)C3)=O)CC2CC1C2NC(c1ccon1)=O C1(C2=CCOCC2)(CNC(Cc2cc(C)sn2)=O)CC1 C(=O)(CC1=CCN(C)CC1)N1CC(CC(C(N2CCC(O)(N(C)CC)C2)=O)F)C1 c12cc3[nH]nc(c3cc1CC)C(=O)O2.N1(C(OCC)OC)CCN(CC)C(C)C1 C1(CNC(C(C)N(C)C)=O)CCN(C(=O)CCc2ccc(O)nc2)CC1(F)F C12(C(N3CC(C(=O)NCCNC(C(CO)OC)=O)C3)=O)CCC(C1)OC2C C1(OCC)CN(C(c2cnc3n2CCS3)=O)C(C)(CNC(C(CC)CC)=O)C1 C1(n2c(-c3ccn(CC)n3)nc(Cc3cc(CC)oc3C)n2)COC2(CCC2)C1 C1(C(=O)NCC2OCCN(CC)C2)C2CCN(C(=O)COC(C)(C)CC)CC12 Cc1oc([N+](=O)[O-])cc1C(N1CCN(C(C2(C)CC(C(C)C)=NO2)=O)CC1CO)=O c1(C(=O)NC(CNC(C(C)NC(=O)NC)=O)CO)ccc2c(c1)CCCC2 Cc1cc(C(N2CCN(C(=O)C(C)O)C(CO)C2)=O)n2nc(C(F)(F)F)cc2n1 c1(C(=O)NC2C(NC(=O)CCc3nc(O)n[nH]3)CCC2)cccc2c1CCO2 c1(C(=O)NC(C2CCOC2)CNC(CCNC(=O)C2CC2)=O)cccnn1 C(=O)(C(C)(O)C(F)(F)F)NC1C(NC(CCN(CCCCC)CC)=O)CCOC1 c1(NC(=O)NCCc2ccc(C)s2)nc(-c2cccnc2)nc2ccccc12 CC(C(=O)N1CC(CN(C)C(c2ccc(CN(C)C)[nH]2)=O)C2(CC2)C1)C(C)(C)C c1(CC(=O)NC(C2(O)CN(C(c3c(C)csc3)=O)C2)C)ccc(Cl)cc1F C1(C(=O)NCC(C)NC(=O)C(C2CCOCC2)C)COC2(CO)CC1C2 N1(C(c2cncc(C)n2)=O)CCC(F)(C(=O)Nc2cn(C)nn2)CC1 c1(C(N2CC(N(S(C3(CC)CC3)(=O)=O)C)C2)=O)ccc(O)c(C)c1O c12cc(Br)c(cc1Br)o2.N1(CC#N)CCC(C2N=N2)C1 c1(C(N(C)CCNC(C2CCC(C)(C)CO2)=O)=O)ccc(O)c2ccccc12 C1(O)(CC)CCCN(CCc2cn(CC(=O)NCC(N3CCCC3)C)nn2)CC1 CC1CN(C(c2ccccc2Cl)=O)CC1NC(=O)CCc1ccc(N(C)C)cc1 N1(C(c2cc(CCCOC)on2)=O)CC2(CCCCN(C(=O)C(C)N(C)C)C2)C1 C1(NC(CC(CC)SC)=O)C(CNC(C2CN3CCN2CC3)=O)CCC12CCC2 C(CCC(C)(C)NC(=O)CCc1cnc(C)o1)NC(C1(C=C)CCC1)=O C12(C)C=CCN1C2=O.c1(-n2cc(CC(c3scnc3C)O)nn2)cccc(N)c1 C1(NC(C23CC(C(F)F)(C2)C3)=O)CCCCC1NC1CCCC(NC(CC)=O)C1 c1(C2C(NC(c3n(C(C)(C)C)ncc3)=O)C2)cccc(F)c1F N1(C(C2(CC)CCCN2C(c2csc(CO)n2)=O)=O)CCCC(F)CC1 C12(C(=O)NCC3(C)C(C)CN(C(CC=CCC)=O)C3)CC1Cc1c[nH]nc12 CCC(C(=O)NCC1(O)CC(NC(=O)Cc2cnn(C(C)C)c2)C1)C(C)C n1(CCC)nccc1C(=O)NC(C)CN(C(=O)CN(c1ccncc1)C)CC c1(C(N(CCCNC(=O)CSCC2CCCO2)C)=O)ccc(F)c(O)c1 C(=O)(C(F)C(C)(C)O)N(c1ccnc(C2CCCC2)n1)C1(c2n(C)nnc2)CC1 c1(C(N(C(CN(C(c2c(OC)ccs2)=O)C)C)C)=O)ccc2nc(C)ccc2c1 C1(NC(CSCC#C)=O)CN(C(C2(Cc3ccc(NC)cc3)CC2)=O)CC1F CC1CC=C(C(=O)N(C2CC(NC(=O)Cc3ccc(C(=O)OO)cc3)C2)C)CC1.O S(=O)(=O)(c1ccc(C)cc1F)NCC(=O)NC1(C=C)CCN(C(C)(C)C)CC1 CCC(C)C(CC(=O)NOCC1CCC1)NC(c1ccco1)=O c1(C(=O)NCC(C)NC(=O)C2=COCCC2)cc2c(s1)C(C)(C)CCC2 C(=O)(C1CCc2cc(F)ccc21)N1CC(CCNC(=O)Cn2ccnn2)(OC)C1 CCCC(C)(CCC)C(=O)N(CCS(C)(=O)=O)CCOC1CCCOCC1 c1(C(C(=O)N(CCCNC(CC(C2CC2)OCC)=O)C)(C)C)ccc(F)cc1F N=c1cc(C(N2CCC(CCCNC(c3cc(Cl)cnn3)=O)CC2)=O)cc[nH]1 N1(C(=O)CCCCO)CCC2(CCCN2C(C2CCCCS2(=O)=O)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CCC(N(C(C(=O)NCC=C)C)CCO)C1 c1(C(N2CCOC(CC(F)(F)F)C2)C(=O)NCC)c(C)nn(C)c1Cl C1(CC=C)(C(=O)NCC(C)(O)CNC(c2ccc(CC)[nH]2)=O)CCCC1 C1(NC(C2CN(CCC)C(=O)C2)=O)CC2CC(NC(=O)C=CC3(C)COC3)C2C1 Cc1ccc(O)c(C(N2CCCC2C(C)NC(=O)COCc2nnc(C)s2)=O)n1 O=C(C#CC1CCCOC1)NCC12CCC(CC1)N(C(C13CCC(C1)C3)=O)C2 Cc1nnc(CCC(=O)NCC2CC2CNC(C2CC=CCC2C)=O)n1C C1(C(=O)NC2C(C)CN(C(c3ccsc3C#N)=O)C2)Cc2cscc2C1 C(=O)(C(C)(C1CCC1)NC(C1CCNC1=O)=O)N(CC#C)CCF c1(C(=O)NC(CC(C)NC(c2cc(C(C)(C)C)c[nH]2)=O)C)cccnc1O c1(C(N2CCC(C)C2CNC(=O)C=Cc2ccoc2)=O)nnc(O)cc1O c1(C(=O)NC2CCC(CNC(COCC=C)=O)C2)ccc(Br)cc1 c1(NC(C2CC3CC3N2C(=O)C=Cc2cnccn2)=O)ccc(Cl)nc1Cl C1(C(N(CCCN(C(c2ccc(COC)s2)=O)C)C)=O)CC2CCCCCC12 CCC(C)C(O)C(=O)NCCN(C(c1ccnc(OCCOC)c1)=O)C1CC1 C1(NC(C(CC)(C)O)=O)CCN(C(C23CCCN2CCC3)=O)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3nncs3)=O)C2)cc1 N1(C(c2c(C)cncc2C)=O)CCC(C)N(C(=O)CCCS(C)(=O)=O)CC1 C=CCC(C)C(=O)NCCC1CC(NC(c2cn(C)c(O)n2)=O)C1 N1(C(c2ccc(COC)s2)=O)CCN(C)CC1CNC(C1(O)CCOC1)=O C1(NC(CCOCC#C)=O)CC(NC(c2cnco2)=O)C(O)C1 c1(OCC)nc(Cl)ccc1S(=O)(=O)Nc1cccc(C2CCCCC2N=[N+]=[N-])c1 N1(C(=O)C(O)C2CCCC2)CCC(C(F)(F)F)n2ncc(I)c21 CC1(C)CCC1NC(=O)CC1CCN(CCC2COCCO2)C1 C1(NC(CC=C)=O)CCN(C(=O)CCC23CCC(CC2)C3)CC(O)C1 c1(NC(C2CCCOC2)CC)ccc(S(=O)(=O)NCc2nn(C)cc2C)cc1C#N c1(C(N(C2CCN(C(c3ccncc3)=O)C2)CC)=O)cc2ccsc2s1 C(CCC(C)C)(C(=O)N1CCCCC1)NC(C1CCC(C#C)CC1)=O C(=O)(CC1=NN(C)C(=O)C1)NC1C=CCN(C(C2(OC)CCOCC2)=O)C1 C#Cc1cccc(C(=O)NCC(C)N(C(=O)CCCn2nc(C)cc2C)C)c1Cl O(Nc1ncnc2c1ncn2CCC1CCNCC1)OC(C)(C)C c1(C(C(=O)NC(CSC)C(=O)O)SC)ccc(Br)cc1 Cc1c(C(=O)NCC2(NC(=O)CCCC(N)=O)CCC2)sc2cccc(F)c12 Cc1cc(C(N2CCCC2C(C)(C)C(=O)NC(c2cc[nH]n2)C)=O)cc(C)n1 C1(CNC(C2CC(CC)C2)=O)CC(C(=O)N(CC(C)C#N)C2CC2)=NO1 C(CC(=O)N1CCC(c2nc[nH]n2)C1)(C(F)(F)F)NC(c1nc(N(C)C)oc1)=O C1(NC(CN(c2ccncc2)C)=O)CC2CN(C(=O)CC(C)(F)F)CCN2C1=O C1(C2N(C(CC=C(C)C)=O)CCC2)CCCN(C(C2CC3(CCC3)C2)=O)C1 Cc1nc(CC(C)C)oc1C(=O)N(CC(C)(C)CNC(=O)CC(C)(O)C1CC1)C c1(NC2CCCC(NC(c3ccc(C(F)F)nc3)=O)C2)ccc([N+](=O)[O-])c(O)n1 C1(CCNC(=O)CCc2cnco2)CCC(NC(c2ccoc2Br)=O)C1 Cc1cnc(NCC2CN(C(c3csc(Cl)c3C(C)C)=O)CC2(C)C)nc1O C#Cc1cncc(C(=O)NC(C)C(C)NC(c2c(C)ccn2C)=O)c1 c1(C(C)NC(C23C(CN(S(C(C)C)(=O)=O)C2)C3)=O)cc2ccccc2cn1 C1C(=O)N=C2C=CN(N2)C2CN1C2.N1(CCO)CCc2sccc2C1.CC(C)CCO N1(C(c2ccc(C(Cl)Cl)cc2)C(=O)NC2CC2)CCC12CCOCC2 C12COCCN1C2=O.Cc1cc(OCC(N2CCCC2)=O)no1.C1CC(=O)N1 C(C(CO)(CO)NC=O)N(C(C(C)OCCOC)=O)C.C(=O)(CCCF)NC N1(C(C2CCN(CC)C2)=O)CC(C(=O)NCCc2cocn2)C(C2CC2)C1 Cc1ccc2c(c1)CC(C(=O)NCCCCNC(=O)C=Cc1ccsc1)S2 CC(Cn1cccn1)C(=O)NCC1(C(=O)NCC2CC2Cl)CC1 Cc1c(Br)c(CNC(=O)Cn2cc(CN3CCN(C)CC3)nn2)nn1C c1(CC)ccc(C(=O)NC2CN(C(c3ccccc3NC)=O)CC23CC3)c(C)n1 c1(CC)onc(C(=O)NCc2cn(CC(=O)NCCc3ccnn3C)nn2)c1C c1(C(=O)NCC2CN(C(C3C4CCCC34)=O)CCO2)cc2c(F)cc(Cl)cc2[nH]1 C1(NC(C2CCOCC2)=O)CCN(C(c2cnn3cnnc3c2)=O)CC12CCC2 C1(C(=O)NC(CCCNC(C=CCC)=O)C)CCC(C)(O)CC1 c1(CCC(=O)NCCOC(C)(C)CNC(=O)C(O)C2CC2)csc(=N)[nH]1 C(=O)(C1=NNC(=O)CC1)N1CCCC(C(C)NC(=O)CN2CCCC2=O)C1 C12(O)CN(CC1O)OC2=O.Cc1ccc(C(=O)COC(=O)OC(C)(C)C)cc1 CC1=NOC(C(=O)NC2COCC2NC(=O)CCF)C1 c1(C(=O)NCC2COCCN2C(C23CCC2C3)=O)cc2c(O)ncnc2cn1 C1(NC(CCSCCNC(C(C)N(C(C)=O)C)=O)=O)CCc2nncn2C1 c1(NC(C(N2CCN(c3cccc(C)c3)CC2)=O)=O)c(C)nc2ccccn12 C1(CNC(CNC(CCC)=O)=O)CN(C(c2cccnc2C2CC2)=O)C2CC12 c1(C(N2CC(NC(c3c(COC)cco3)=O)C(C)C2)=O)ncn2c1CCCCC2 C12(NC(c3nc(COC)sc3)=O)CCCN(C(c3cccs3)=O)CC1C2 N1(CC(=O)NC(c2cn(CC(=O)NCC)nn2)(C)C)C(=O)CC(C)(C)C1=O N1(C(C2C(CNC(CC)=O)C2(C)C)=O)CCC(F)(F)CC1 C1(CC=C)(C(=O)NCC2(c3ncco3)CC2)CCN(C(C2CC(=C)C2)=O)C1 c1(OC)cc(OC)nc(N2CCCC2CNC(c2cc(F)cc(F)c2)=O)n1 CC(C)CC(F)C(=O)NCCOCCN(C(=O)CC1CCCCC12CC2)C C(=O)(CCC(C)(C)C)NC(C1CCN(C(c2c(C)scn2)=O)CC1)C N1(C(C(CSC)O)=O)CCCC2(CCN(C(C3(CC(C)C)CC3)=O)C2)C1 N1(C(CCc2onc(C(C)C)n2)=O)CC2(CCN(C(C3CNC(=O)N3)=O)CC2)C1 c1(OC)c(C(=O)N(C)CC2(O)CCN(C(C3(CC(C)C)CC3)=O)C2)ncnc1C C(CC(=O)NC1CCSC1)(C(F)(F)F)NC(c1nn(C)c(=O)cc1)=O CC(CCC(=O)N1CC=CC1Cn1cc(-c2nccn2C)nn1)N(C)C C1(NCc2ccc(N3CCN(CC)CC3)cc2)CCCCC2(CC2)C1 c1(C(N2CC3CN(C(c4nn(C)c(F)c4)=O)CC3C2)=O)cccc2cnccc12 C1(NC(COCCCOC)=O)C=CCCC1C(=O)NCCCCSC CC(C)CC(C(=O)NOCCOC(C)C)NC(=O)CC1CC1(C)C N1(C(C2(CCCC)CCCC2)=O)CC(NC(=O)C=Cc2cc[nH]n2)CC(F)C1 N1(CCC)CCC(CNC(=O)CCN(C(=O)C(C)NC=O)C(C)C)C1 C1(NC(CN(C)C(N)=O)=O)CCN(C(=O)Cc2cc(Cl)sc2Cl)C1(C)C C1(NC(C(C)N(C(=O)COCC(C)C)CCC)=O)CCCN1 Cc1ncnc(O)c1C(N1CCC(O)CC1)C(=O)NCc1cccc(Cl)c1 CC(C)(C)CC(C(=O)NCCOC(=O)C1CC1)NC(C1CC=CCC1)=O C(=O)(C(C(C)NC(=O)CN(C)C1CC1)C(C)C)Nc1cccc(OCC)c1 C(=O)(CC1OCCc2sccc21)NCCN(C(c1c(C)c(Cl)cnc1)=O)C1CC1 N1(C(CCOCC(C)C)=O)CCN(C(C2(CF)CCC2)=O)CC1 C1(C(=O)NCCC(C=C)C)CN(C)CCN1C(c1cnncc1NC)=O CC1(C)C(=O)Nc2ccc(C(N3CC(NC(c4ccco4)=O)CC(F)C3)=O)cc21 C(c1ccco1)=CC(=O)NCC1N(C(C(n2ccc(C3CC3)n2)C)=O)CC1 C(=O)(CC(C)(C)N(C)C)N1CC(OCC(=O)N(C)CC2(O)CCOC2)C1 Cn1cccc1C1CC1C(=O)NCCNC(c1csc(-c2cnccn2)n1)=O N1(C(C2N(C)C(=O)NC2)=O)CC23CCCC2(C1)CN(C(C1C=CCC1)=O)C3 N1(C(C(COC)OC)=O)CCC(NC(=O)CNS(N)(=O)=O)C(O)C1 c1(OC)ccc(C(C)=CC(N2CCCN(C(c3ccoc3)=O)C(C)C2)=O)cc1 N1(C(c2cc(C)n(-c3ccccc3)n2)=O)CCC2(C1)CN(C(=O)C=CCO)C2 CC1(C)CN(C(c2cc(C#N)c[nH]2)=O)CC1C(=O)NCCC(O)CCO O=C(N=c1[nH][nH]c2cccnc12)C(=O)N1CCN2CCS(=O)(=O)CC2C1 N1(C(C2CC(CNC(C3N(C)CC(C)(C)C3)=O)OC2)=O)CCC2(CC1)CN(C)C2 C1(C(=O)NC(C)CNC(=O)CCc2cccs2)CCC2(CC1)CC2 CCC(CC)C(F)C(=O)NCC(=O)NC1CC(C)(CNC(c2ccoc2)=O)C1 CCCC(C)CC(=O)N1CCC(N(C)C(c2cnn(C3CC3)c2)=O)C1 C(=O)(C1=Cc2ccccc2C1)NC1C(C(=O)NCC2CC3(CC3)CO2)CCC1 C1(NC(C(CC)(CO)OC)=O)CC12CCN(C(=O)CCn1ncn(C)c1=O)CC2 C1(NC(=O)Cn2ccnn2)CN(C(C2CCCOCC2)=O)CC1n1cccn1 CC1(C)CCCC(O)(CNC2CCCCCC2C(F)(F)F)C1 CC(C(=O)NCC1CCCCN(C(=O)CCC(=O)c2cccnc2)C1)S(C)(=O)=O C1(NC(CN(C2CC(OC)C2)CC(C)C)=O)CC(C)(C)CO1.C(C(=O)NC)OCC c1(CC(=O)NCC2(C)CC(NC(C3CCC(=O)N3)=O)C2)cn2ccccc2n1 C(c1ccc(O)c(O)c1)=CCNC(=O)NCC=C.CC1CC1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(C2CC3CCC(C2)S3)=O)CC1(C)C c1(C(N2CCCCC2)=O)cn(CCNC(C2(C3CCCO3)CC2)=O)nn1 O=[N+]([O-])c1cccnc1N1CCOCC(COCc2ccccc2)C1 c1(-c2cc(NCc3nc(C)oc3)ncc2)cc(O)c2ccoc2c1 N1(C(c2ccc(NC(c3c(C)cnnc3)=O)nc2)=O)CC2CC2C1C#N C1(C(=O)NCC2C=CCOC2)(CC)CCN(C(=O)C(O)Cn2cncn2)C1 CCCC(C)C(=O)N1CC(SC)C1.c12ccc(cc1)-c1cn(nn1)C2 C1(C(C)C)CCN(C(=O)C(N2CCCC(Cc3nccn3C)C2)=O)CC1 c1(C(C(N2CC(=CC(C)NC(C(C)OCCOC)=O)C2)=O)C)cccc(F)c1 c1(CCC(c2n(C(C(=O)OC)C)nnn2)(C)NC(C)(C)CSC)cccc(Br)c1 N1(C(C2(CC)CC(C)(C)C2)=O)CCC=C(CNC(c2n[nH]cc2C)=O)C1 C1(NC(=O)C2=CCSC2)CCN(C(c2csc(Cl)n2)=O)C(c2ccccc2)C1 N1(C(c2ccc(CCC)s2)=O)CCCC(N(C(C2CC(C)(O)C2)=O)CC)C1 c1(-c2nnc(CCC(=O)OCC(N(OCC)C)=O)o2)ccc(C#N)cc1OC N1(C(CC(CNC(C(C)CC(F)(F)F)=O)(C)C)=O)CCC2(COC(=O)N2)C1 c1(SCC)cc(Cl)ccc1C(=O)NCC(C)CNC(=O)COCCF C1(CC(=O)NC(CC#C)CC)C2CCCC2N1C(=O)CC1(C#N)CCOCC1 C(C(C)(C)CNC(=O)C(F)CC1CCCCC1)N(C(=O)C(F)n1cccn1)C C1(OC)CN(C(=O)CCc2ccsc2)CCC1CNC(=O)C(C)(C)COC Cc1ccc2[nH]c3c(c2c1)CC(NC(N1CC(O)CC1(C)C)=O)CC3 Cc1ccc(C(N2CC(OCCNC(=O)CC3CCCCC34CC4)C2)=O)nc1O CC1(O)CCC(C(=O)NCc2cc(C(N3CC4(CC4)CC3CO)=O)co2)CC1 N1(C(c2cc(C)nn2C)=O)CCC(NC(=O)C(c2ccccc2)O)C(F)C1 CC1OC2(C(=O)NC(c3cccc(Br)c3)CC3CC3)CCC1CC2 c1(Cc2ccc(C)c(NC(C3CC3)=O)c2)nnc2c(Cl)cc(C(F)(F)F)cn12 CCC(CN1CCCC(c2n[nH]cc2OC)C1)CC(F)F N1(C(CCc2n(C)cnn2)=O)CCCCC1CCNC(C1CC2CC2C1)=O C1(NC(C2(C)CCN(C(CN3C(C)CCC3)=O)C2)=O)CC(C)CCC1O n1(C(C)C)cc2c(n1)CC(C(=O)OCC1CCOCC1(C)C)CC2 CC1C(NC(=O)CCNc2ccccn2)CCCN1C(c1ncc(F)cn1)=O C(=O)(C1COc2c(C)cccc21)NC1C2CN(C(CCC(=O)NCC)=O)CC21 CC1(C)CCc2cnc(C(=O)Nc3cncc4c3CCC4)nc21 N1(C(CNC(CCC)=O)=O)CCC2(CCN(C(c3ccc4ccccc4c3)=O)C2)C1 c1(N2C3CC(NC(C4(CC)CCC(O)CC4)=O)C2CC3)ncnc2[nH]ccc12 N1(CC(=O)NCC(O)CCNC(c2cncc(Br)c2)=O)CC2CCC1C2 C1(C(=O)NC2CC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)CCn2ncnc2C1 C1(CC)(CC)CCN(C(=O)C(C)N(C(=O)C(CC2CC2)OC)C)C1 C(=O)(C1=COCCO1)N1CCC(N(CCC)C(C2CCC2C#N)=O)CC1 Cc1nc(N(C)C)sc1C(N1CCC(CN(C(=O)C=Cc2ccncc2)C)C1)=O N(C(=NCCC1CC(C(F)F)C1)NC(C)C)CCCC C1(NC(c2ccc(CSC)o2)=O)CC(C)CN(C(=O)COCCN(C)C)C1 CC1CCCC(O)(C(=O)NCC2(NC(c3ccsn3)=O)CCC2)CC1 N1(C(Cc2c(C)nccc2)=O)CC(NC(c2cncc(CO)c2)=O)CC2(CC2)C1 CCC(C(=O)N(CC(C)NC(c1cc(C(C)C)ccc1C)=O)C)C(C)(C)CC C1(C(N2CCC(NC3CCN(C)C3=O)CC2)=O)CCC2(CC1)CC(N(C)C)C2 Cc1ccc(N)c(C(=O)NCC(C)CNC(=O)Cc2cnc3n2CCCC3)c1F CC(C)(O)C(F)(F)CNC(=O)Cc1csc(NC(C2CCCC2)=O)n1 C(CC(C)(C)C)(C(=O)NCC1CCN1C(C1(C#N)CC2(CC2)C1)=O)OC c1(C(=O)NC2C(NC(c3cc(C)sc3)=O)CC2)c(C)noc1C(C)C CC1(CNC(=O)CS(c2n[nH]c(=N)s2)=CCl)CCCN(C(C2(C)C=CCCC2)=O)C1 Cc1ccc2nc(C)cc(C(=O)NC3CCC(N(C)C(c4cn[nH]c4)=O)C3)c2c1 C(C(C)C(=O)NCCCCN(C)C(c1cc(C(N)=O)c[nH]1)=O)N(CCCOC)C c1(CCC)nc(C(O)Cc2ccccc2F)n(-c2cnn(C)c2)n1 C12(CNC(CC=CC=C)=O)CN(C(=O)CSc3cccs3)CC(F)(C1)C2 c1(OC)ccc(C(=O)NC(C)CCNC(=O)Cn2c(C)ccc2C)c(F)n1 C(=O)(C1=CC(O)C(NC(=O)C(C)=CC(C)(C)C)C1)N1CC(CCO)(CC)C1 C1(C(=O)NC2(CO)CCCN(C(=O)C3=CCC3)C2)CN2CCCN1CC2 N1(C(C(CC=C)C)=O)CCCC(CNC(c2cc(CC)ccc2Cl)=O)(OC)C1 Cc1nccc(C(N2CCCC(C(=O)N(C(=O)Cc3ccno3)C3CC3)C2)=O)n1 Cc1cc(C(N2CCOC(CN(C)C(C3CC4(C3)CC(C)C4)=O)C2)=O)cc(C)n1 C1(C)(NC(C(C2CCCC2)OC)=O)CN(C(=O)C(C)=C(C)C)C(C)(C)C1 C1(C(N2CCC(CNC(c3cc(OC)cc(C)c3)=O)C2)=O)CCn2nncc2C1 N1(C(c2cc(Cl)cc(Cl)c2)=O)CC2CCC1CN2C(C1CC2CC12)=O c1(CC(N2CC(N3C(=O)CC(NC(C=CC=CC)=O)C3)C2)=O)ccc2[nH]ccc2c1 Cc1nc(C(F)(F)F)oc1C(=O)NC(C1CCCN(C(=O)Cn2cnnn2)C1)C C1(OC)CC(CNC(c2ccc(O)cn2)=O)N(C(c2ccc(CO)nc2)=O)C1 c1(SC)nccc(CNC2CC(NC(c3cc(C(F)(F)F)ccn3)=O)C2)n1 CC1CCc2n[nH]cc2C1C(=O)NCCN(C(c1cc(CO)on1)=O)C1CC1 c1(NC(C2CC(Nc3nccc(OC)n3)C2)=O)cnn2cccnc12 C(=O)(N=c1[nH]nc(-c2cccc(Br)c2)s1)N(CCCNC)Cc1ccccc1 Cc1cncc(C(N2CCCC2C(C)(C)C(=O)NC(C)CS(C)=O)=O)c1 c1(C(=O)NCC(CC(C)C)NC(CCC(C)=O)=O)c(F)ccc(C)c1Cl C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CN(C(=O)C(C)(C)C(F)F)CCC1CO Cc1nc(N2CCCCC2)sc1C(=O)NCCC(=O)NCC1CCC1 C(CCCC(=O)NOC(CO)C(C)C)N(C(C(CCOC)(C)O)=O)C N1(C(C(CC)C)=O)CCC2CCC(C1)N2C(c1c(F)ccc(C#N)c1F)=O C=C(CC)CN=c1nc2c(ncn2C(C)C)c(NC(C)CN2CCCOCC2)[nH]1 c1(C(N(CC(C)NC(c2ccn(C)c2)=O)C)=O)c(Cl)ccc(Cl)c1N c1(N2CCCN(C(CCSC)=O)C(C)C2)ncnc2ccc(O)cc12 C(=O)(C(F)C(C)CCC)N(c1ccccc1)C1CC1.C1(=O)C(COC)CN1 C1(CC(=O)NC2CCC(CNC(C34CC(C)(C3)C4)=O)C2)(OC)CCCCC1 C1(C(=O)NC(CC(=O)NC)C2CC2)CC(=O)N(C(C)(C)C)C1=O CC1CCn2ncc(C(=O)NC3CCN(C(c4n[nH]c(=N)[nH]4)=O)C34CCC4)c2C1 Cc1c(C(=O)NC2CC2CNC(=O)C(F)=CCCF)cnc2ncnn12 C(=O)(N(CC)OC)c1cn(CC2N(C(=O)NC(C(=O)NC)CC)CCC2)nn1 N1(C(C(C)CC(N)=O)=O)CCC2CN(C(=O)CCOc3ccccc3)CC2C1 c1(C(=O)NC2C3CC(O)C2N(C(=O)C=C2CCC2)C3)ccc2c(c1)COCC2 c1(C(=O)OC)c[nH]c(=NC2CCCC(NC(=O)CC3COCCO3)C2)cn1 CCS(=O)CC(=O)N1CC(C)(CCC(=O)NCC(C)(COC)OC)C1 n1(CC)nc(C)c(C(=O)NC2COCC2NC(C2(OC(C)C)CCC2)=O)c1Cl c1(COC)sccc1C(=O)NCC(CNC(=O)C(c1cccnc1)OC)CO S(=O)(=O)(c1cccc(CN)c1)Nc1c(=O)cc(C(=O)OC)n(C)c1 C12(C(=O)NCc3nc(OCC)oc3)CC(C)(CN1C(c1cnc(N)cn1)=O)C2 C1(NC(C(C)OCC=C)=O)CN(C(c2cn(CCOC)nn2)=O)CC1O C#CCCCC(c1nnnn1CC(=O)OCC)NCC(CO)SCC(F)F c1(C(=O)NC(C)CNC(=O)Cc2csc(C3CCOC3)n2)cccn2ccnc12 C12(C(N3CCC(NC(C4OCC5CCCC45)=O)(CF)C3)=O)CC3CC1C2C3O N1(C(Cc2ccc(C)s2)=O)CCC2CCN(C(c3cc(C(F)F)nn3C)=O)C2C1 N1(C(CN(C)CCO)=O)CCCC12CCN(C(c1ccc(O)nn1)=O)C2 C1(CNC(c2c(C)nncc2)=O)CN(C(C2CC2C(C)O)=O)CCN1C C1(C(=O)NC2CC(OC)C2)CCC(CNC(c2cscc2Cl)=O)CC1 c1(N2CCCC(C(N3CCCCC(NC)C3)=O)C2)nc2cc(C)cc(C)c2s1 C(=O)(C1=C2CCN=C2NC=C1)N1C2CC(CN(C(C3(C)CC3Br)=O)C2)C1 CC1CC(C(N2CCN(C)CC2)=O)CCN1C(=O)CS(=O)(=O)N(C)C C1(c2cn(CC(=O)NCC(C)N(C(=O)C3CC3)CC)nn2)CC(F)(F)C1(F)F c1(C(N(C2CCN(C(COCC=C)=O)CC2C)C)=O)ccc(Cl)c2ncccc12 C12C=CC(C1)N2.c1(C=O)cccs1.C1(N(C(C)C)C)(C(=O)NC)CC1.C(=O)(CSC)N c1(C(N2CC(NC(C(=O)N(C)C)=O)CC(C)(C)C2)=O)cc(Br)cc2[nH]ncc12 C(=O)(C1CCCc2cccnc21)N1CC(OC)(CNC(C2CC(=O)CO2)=O)C1 C(=O)(C1=NOC(C)C1)N1CC(C)(NC(c2cnn(CC)c2C)=O)C1 CCC(O)CC(=O)NCCC(C(=O)NCCC1CCN(C)C1)OC C(=O)(CC(C)(C)C(F)F)NCC(CNC(C1CCCN(C(=O)OC)C1)=O)OC C1(C(=O)OC)C=CC1C(N1CC(CNC(=O)CC2(C(F)F)CC2)C1)=O c1(C(N2CCCC(CC)(NC(C3CC(SC)C3)=O)C2)=O)ccc(F)c(OC)c1F N1(C(C(COC(C)=O)C)=O)CCC(C2CC2)C1Cn1cc(CN2CC3CC3C2)nn1 O=C(CCCC1CCCO1)NCC(O)C(=O)NCCc1ccncn1 C1(C(=O)NC(CO)CCO)C=CCN1C(c1cc(Cl)ns1)=O C(=O)(CCCCCCCCCO)NCC1N(C(c2c[nH]c(=N)o2)=O)CCCCC1 C1(C(=O)OC)CC(F)(F)CC1C(N1CCC(O)(CNC(=O)CN(C)C(C)C)C1)=O CC1CC2CN(C(C3CCC4(CC4)N3C(c3cc(CO)on3)=O)=O)CC12 C(c1ccc(F)cc1)=CC(N1CC2CC1CN2C(C1(F)CCCC1)=O)=O C(=O)(CC(C)C1CCCCC1)NCC(CC)NC(C1CCCCO1)=O C1(C(=O)NN(C)C)CCN(c2nccc(O)c2)CC1O.N1(C(C)C)CCC(C)CC1 C1(NCC(C2CCOCC2)OC)CC(NC(c2csc(Cl)c2Cl)=O)C12CCC2 CCC(CC)(CCNC(C1CN(C)C1)=O)NC(C1CCN(C2CC2)S1(=O)=O)=O CC1(C)Oc2ccc(NC(c3c(F)cc(Br)cc3Cl)=O)cc2O1 c1(C(=O)NCCCOCCN(C(C2CC(CC)C2)=O)C)cccc(Cl)c1F C1(NC(c2c(C)[nH]nc2Cl)=O)COC2(CNC(=O)C=CC(F)(F)F)CC1C2 Cc1nc(C(C)C)sc1C(N1CC(CNC(c2csc(C3CC3)n2)=O)CC1C)=O CCCS(=O)(=O)CC(=O)NC1COCCN(C(=O)CSCC(=O)OC)C1 C12(CNC(C(F)=CC)=O)CCCC1N(C(=O)COCP(C)(C)=O)CCC2 C(=O)(CC(C)(C)CCC)NC(CC=C)CNC(=O)C(C)S(C)(=O)=O c1(C(N2CC(F)(C(=O)OC)C(F)C2)=O)sc(S(N)(=O)=O)c(OC)c1OC N1(C(CNC(C(C)(C)C)=O)=O)CC(NC(=O)C2=C(Cl)CCCC2)CC(F)(F)C1 CC1=C(C(=O)N2CC(NC(c3csc4nccn34)=O)CC2(C)C)COCC1 c1(C(N(C2CCC(C)C2)C)=O)cc(Br)cn2ncnc12 c1(C(=O)NCC(CNC(C(CCO)N(C)C)=O)CO)ccc(Cl)c(N)c1 Cc1cnnc(O)c1C(N1CC(C(=O)NCC2CCC2(F)F)CC(C)C1)=O c1(SCC(=O)NC23CC(NC(N4CCCCC4=O)=O)(C2)C3)cccnc1C(C)(F)F c1(CN(C2CCOCC2)CC(=O)Nc2nc(C)on2)cc(Br)c(F)cc1C CC1(C)CC(CNC(=O)C=Cc2ccco2)N(C(C2CC=CCC2)=O)C1 N1(C(c2c(Cl)csc2Cl)=O)CC2(C1)CN(C(C1(CO)CCC1)=O)CCO2 c1(OC)c(C(=O)NC2CC23CCN(C(c2cnsc2)=O)CC3)cccc1[N+](=O)[O-] Cc1ccc(C(C)NC(N2CCC(Nc3ncccn3)C2)=O)s1 c1(C(=O)NCCCn2c(C)nnc2)ccnc(OC2CCN(C(C)C)C2)c1 Cc1cocc1C(=O)NCC(c1ccccc1)N(C(=O)Cn1nccn1)C Cc1cc(F)sc1C(=O)NC1CCCC1CNC(c1csc(Cl)c1Cl)=O C1(=CC(=O)NCC2C(CC(=O)NCCCCOCC)C2)CCCCC1 N1(C(c2c(Cl)cc(C)nc2)=O)CCCC2(CCC(NC(=O)CCC(C)C)C2)C1 C1(NC(=O)C(N2CCCCC2c2ccc(F)cc2)=O)CC2(CCNC2)C1 C(CC)(CC(F)F)CNC(CN(C(=O)Cc1ccc(C)cc1)CCC)=O C(C(C)(C)CN(C(=O)COCCCF)C1CC1)N(C(=O)CC1CCC2CC12)C N1(C(C(C)Cc2ccccc2)=O)CCCC2C1CCN2C(C12COC(C)(C1)C2)=O c1(CCC(N2C(CNC(C3C(CC)CCO3)=O)CCC2)=O)ccc([N+](=O)[O-])cc1 C(CCC(C(=O)N1CC(c2ccco2)C1)NC(=O)C(C)CSC)OC C1(NC(c2cnon2)=O)CCCN(Cc2ncc(-c3cccc(F)c3)o2)C1 c1(CNC(=O)C(=O)NC2C3CN(C(C(CCC)C)=O)C2C3)c(Cl)cccc1Cl c1(CCNC(CN(CC#C)C(c2ccc(CC)s2)=O)=O)ccncc1F C1(C(=O)NC2CC(NC(c3cnc(CC)[nH]3)=O)C2)C(C(=O)OC)CC(=O)N1C c1(CN(C(=O)C(C)(C)C)C)cnn2c1CN(C(=O)CCc1ccncc1)CC2 Cc1cc(-c2ccccc2)oc1CC(=O)NC1(CNC(=O)CC2(C)CC2)CC1 c1(-n2cc(C(=O)NCCCC(C)(C)NC(=O)C(C)(C)F)nn2)ccc(Cl)cc1Cl Cc1ccc(CC(=O)NCCCCC(C)NC(c2cn(C(F)F)cn2)=O)c(C)c1 C(=O)(CC(CNC(=O)Cc1ccsc1)OC)N(C(CC)CC)CCO C(C)(C)(CN=c1nc(SC)[nH]s1)C1CN(C(c2ccn(CC)n2)=O)C1 CC1CN(C(c2cn(C3COC3)nn2)=O)C(C)CN1C(=O)COCC1CC1 c1(C(N(C(CCNC(C2(CC(C)C)CCC2)=O)C)C)=O)nnn2c1C(=O)NCC2 C(CC(C)(C)C)(C(=O)N1C(CC(=O)NCC(N2CCCC2)C)C2CCCC12)OC c1(CC(=O)NC(COC)C(=O)NCc2cocn2)cncnc1O C1(C(=O)NCC(C)CN(C(=O)CCC2OCCO2)C)CCCC(F)(F)C1 c1(C(=O)NC(CCSC)C(=O)NCc2cc(C)cs2)cncc(F)c1C C1(CNC(Cc2nc(CC)sc2)=O)CN(C(=O)C(CSC)OC)CC1C(F)(F)F N1(C(c2cc(C)[nH]n2)=O)CC2CC(C)N(C(=O)C(C3CCC3)C3CCC3)C2C1 C1(NC(C(=O)Nc2c(C(=O)OC)cccn2)=O)CCNCCC1CO CCN=C(NCc1cc2c(cc1OC)CC(C)O2)N1CCCC(Cn2ccnn2)C1 c1(CC(=O)NC(CNc2cc(COC)ncn2)CC(C)C)nc2c([nH]1)CCCC2 c1(C(N(CCCNC(c2coc(Br)n2)=O)C2CC2)=O)cc2ccccc2cn1 c1(C(CO)NC(C2C(C(C)NC(=O)C(F)n3ccnc3)C2)=O)cnn(C)c1 C(=O)(CCCCC(=O)NC1CC(F)CN(C(c2nccn2C)=O)C1)OC c1(C(=O)NC(CNC(Cc2c(C)n(C)nc2)=O)C(C)C)coc2c1COC2 C1(CC(=O)NC2(CF)CCC2)CCN(Cc2cnc[nH]2)C1 Cc1cc(C)n(Cc2nc(Cc3ccccc3F)nn2CC(N)=O)c(=O)n1 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCCC(C)(C)C1CNC(C1CC1CF)=O N1(C(C2(C(C)C)CC2)=O)CCCN(C(c2nocc2C2CC2)=O)CC1CO N1(C(C(CSC)O)=O)CC2(NC(c3ccoc3C(C)C)=O)CCC1CC2 c1(OC)ccc(F)cc1C(=O)NCC(C)(CO)NC(=O)CC1CC2(CCC2)C1 c1(C(=O)NCCCCn2cc(-c3cc(C#N)[nH]c3)nn2)ccc2c(c1)CC2 C(C(=O)NCC(C)(C)NC(c1occc1Cl)=O)(C(C)C)c1cnc(C)s1 CN1C(=O)CCC1CC(N1CCCCC1C1(NC(=O)CSC2CC2)CC1)=O C(=O)(C(C)CC(N)=O)NCCC1(OC)CN(C(=O)CN2CCC2C)C1 Cn1nc(C(=O)NCc2csc(CNC(c3cnoc3C3CC3)=O)n2)cc1O c1(OC)ccccc1CCC(=O)N1CC(C(C)NC(=O)CSCC(N)=O)C1 C1(NC(COCCC)=O)CN(C(=O)Cn2nccc2N)C2CCCCC12 CC1(CNC(c2cocn2)=O)CCCN1C(=O)CC1CCCNC1=O CN1CCC(C(=O)NC2CC3CC2N(C(c2nnc(S)n2C)=O)C3)S1(=O)=O C1(C(=O)NC2(CC)CCOCC2)CC2(C1)CN(Cc1cccnc1F)C2 N1(CC(=O)NCC=C)CC(C(=O)O)C2(CN(C(c3cc(F)c(Cl)nc3Cl)=O)C2)C1 c1(C(=O)NC(CCC)CNC(c2cc(C)sn2)=O)cnc2cccc(C)n12 C1(C(N(C)CCN2CCN(C(C3(C(C)(C)O)CC3)=O)CC2)=O)CC2(CCC2O)C1 C1(CC(=O)OC)CCCN(N2CCC(Cc3ccc(F)cc3)C2)C1 CN1CCN(C(C2C(C)(C)C2(C)C)=O)C(C(N2CCC(C(C)(C)O)C2)=O)C1 N1(C(c2n(CCOC)ncc2)=O)CCCCC(CNC(=O)C(F)=C2CCC2)C1 c1(C(N2C(CCNC(CCC(C)OC)=O)COCC2)=O)cc[nH]c(=N)c1[N+](=O)[O-] CN1C(=O)CCC1C(=O)NCC(C)(C)NC(=O)C(C)NC(C1(CO)CCCC1)=O c1(C(=O)NC2C(NC(c3c(C)ncn3C)=O)CC2)ccc(F)c(F)c1F c1(SC)cc(C(N2CCOC(C(C)NC(=O)C=C(C)Cl)C2)=O)ccc1NC(C)=O Cc1cccc2c(C(N3CCC(N(C)C(c4nc(O)[nH]c(=O)n4)=O)C3)=O)coc12 C(=O)(CCS(N)(=O)=O)NCC(CC)(CC)NC(c1cn(CC)nc1C(F)(F)F)=O N1(C(c2c(CC#N)cccc2)=O)CCC(O)CC1C(=O)NC1CN2CCC1CC2 c1(NC(c2c(-c3c(C4CC4)cccc3F)cncc2F)=O)cccn2nccc12 N1(C(Cc2nc(C)c(C)[nH]2)=O)CC2(CCC(NC(c3cc(C#N)on3)=O)CC2)C1 C1(NC(c2n[nH]c(CC)c2C)=O)CCCC(C(=O)N(C)Cc2n[nH]c(C)n2)CC1 C(C)(C)(CCCCC(=O)N1CCCC(CN(C)C(c2cccc(O)n2)=O)C1)OC CC12CCC(C(N3CC4CCCC3C4CNC(=O)C3=CCC3)=O)(CC1)CO2 C(=O)(C(CNC(C1(C)CCCC1O)=O)CC1CC1)NCC1(C)CCC1 C(=O)(CC(C)C(=O)OCC)NCCC(=C)CNC(c1ccnn1CC)=O c1(-n2cc(CCNC3N(C(C(C)SCC)=O)CCC3)nn2)cc(C)cc(F)c1 c1(SC)cc(=NC(=O)C2CC=CC(NC(C3CC3(C)C(F)F)=O)C2)[nH]n1C C#Cc1cncc(C(=O)Nc2ccccc2C(=O)Nc2cc(F)ccc2OC)c1 Cc1coc(C(=O)N(C2CCCC(CCn3cccn3)C2)N2CC(C)(C)C2)c1C c1(N2CC(NC(C(=O)NC(C)C)(C)C)C(C)CC2)ncc([N+](=O)[O-])cc1Br c1(OC)nc(C)ccc1C(=O)N(CC(C)O)CCNC(=O)CCc1nccs1 c1(C(=O)NC2CC(CCNC(C3CCC(C)(CC)O3)=O)C2)ccc(OC)c(N)c1 O=C(C1CCCn2cnnc21)NCC1COCCN(C(=O)C(F)CC2CC2)C1 C1(C(c2n(CCOC)nnn2)NC2(CSC)CCC2)CC2(C1)CC(O)C2 C(CCS(N)(=O)=O)NC(C(=O)NC1C(CC(=O)N(C)CC2CC2)CCC1)=O N1(C(c2nnc(C)s2)=O)CCC(F)(CNC(C2(C(C)C)CC2)=O)CC1 C(c1ccc(F)cc1)=CC(=O)NCC(C(C)C)NC(c1cccc(C#N)n1)=O N1(C(C2C(=C)C2)=O)CCc2c(c(CNC(=O)CCc3cccnc3)nn2C)C1 c1(C(=O)NCC2CC(NC(CC3(C)CCC3)=O)C(O)C2)cc(C#N)ccc1Cl c1(C(=O)NC2(CCNC(C=C(C)C3CC3)=O)CC2)csc2c1CCC(C)C2 N1(C(CNC(CCCCC)=O)=O)CC(NC(c2ncn(C(C)C)n2)=O)CCC1C CCCN=C(NCc1cn(C)nc1-c1ccccc1)NC(C)CC C1(CCNC(CCC2(C)CC2)=O)CN(C(c2cnn[nH]2)=O)CCS1(=O)=O N1(C(C2(OCC)CC2)=O)CC23CCCCC2(C1)CN(C(=O)CNS(=O)(=O)NC)C3 CCC(C(=O)N1CC(CC(=O)NC(C)CN=[N+]=[N-])(OC)C1)n1cncn1 Cn1nc(CNC(=O)C#CCNC(C2CCCC(F)C2)=O)oc1=O N1(C(CC=CCCCC)=O)CCCCC(NC(=O)CCCC(C)=O)C1 c1(C(=O)NC2CCN(C(C(C(=O)OCC)OC)=O)C2CC)cccn2nccc12 C(CC(=O)NCC1CC1NC(C1(C(N)=O)CC1)=O)(C(C)C)OCC c1(OC)ccc(F)cc1C(F)(F)C(=O)NC(CNC(=O)C=C(C)Cl)CC(F)(F)F CCC(C(=O)N(C)CCNC(=O)C=C(C)C(C)C)NC(=O)OC(C)(C)C c1(CC)nnc2cc(NC3CC(NC(=O)CC4CC(C)(C)CO4)C3)ncn12 C1(C(=O)NC2(C)CC=CC2)CCN(C(=O)C(O)C(F)(F)F)C(C)(C)C1 C1(C(=O)NCC2N(C(C3CCOCC3)=O)CCC2)CC2C=CC1O2 C(CC(=O)N1CC(C#N)(SC)C1)(C(C)OC)NC(c1ccc(OC)o1)=O CN(Cc1ccc(OCC(=O)O)cc1)N1CCc2c(cnn2C)C1 c1(C(C)C)nc(NCCC(C)C(C)C)cc(=NC2CCCn3cnnc32)[nH]1 C1(N(C)C(C2CC23CCCC3)=O)CN(C(c2cnc(C3CCC3)o2)=O)CC1(C)C C(CN=c1[nH]cncc1I)C1CCC(NC(c2ccoc2Cl)=O)C1 C1(C=C)(C(N2CCC(N(C(=O)CC3COCCO3)CC#C)C2)=O)CCCCC1 c1(C(N2C(CNC(C=C(C)C)=O)CCC2)=O)cnc2c(c1)c(=O)n(C)c(=O)n2C N1(C(C(C)n2cccn2)=O)CCN(C(=O)C2=COCC2)CC1c1ccccc1Cl Cc1cc(-c2noc(C(C)NC(C)C(C)CCN(C)C)n2)c(C)o1 C1(CN(C(=O)C(F)C2CCC2)C)COCCN1C(c1ccnc(CO)c1)=O CCCCCC(CC)C(=O)NC1(C2(COC)CCCCC2)CC1 C(=O)(C(F)CC1CCCCC1)NCC(Cc1ccccc1)NC(CN(C)CC)=O N1(C(C(CC(C)C)F)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 C(=O)(CC(C)(C)CCOC)N1CCC(N2CCN(C(CCCCOC)=O)CC2)C1 c1(OC)ccc(C(CNC(=O)NCCC2CCOC2)CO)cc1OC CS(C)(=O)=NCC(=O)N1CCN(C(=O)COCC2CCCO2)CC1CC(F)F c1(C(=O)NCCC(C)NC(=O)C2Cc3ccccc32)nnc(O)c2ccccc12 c1(NC(N2CC(C3OCCC(N)C3)C2)=O)ccc(S(=O)(=O)NC2CC2)cc1 c1(C(=O)NCCC2CC(NC(CC(C)c3ccco3)=O)C2)csc([N+](=O)[O-])c1 C1(NC(COc2ccc(C)cc2Br)=O)CCCCN(C(=O)C#CC2CC2)CC1 CCC(CC(=O)NCC1CC2CCC(C1)N2C(c1ccoc1C1CC1)=O)C(C)C n1(CCNC(c2cnsc2)=O)cc(C(=O)NC2(CO)CC(F)C2)nn1 C(=O)(C1=CCCN(C(=O)CN)C1)NC(CCSCC)C.C(=O)(NC)OC N1(C(c2c(C)noc2-c2cnccn2)=O)CCC(C)(C)C(NC(=O)CC(F)F)C1 c1(C(=O)OCC(CSCC)(C)C)c(OC)cccc1O Cc1cc(F)cc(C)c1C(=O)NCCCc1cn(-c2cccc(Br)c2Cl)nn1 C(=O)(C(CO)C(C)(C)C)N(C1(c2c(C)nsc2)CC1)C(=S)NC(C)C(=O)N(C)C N1(C(C(CC)C)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC12CCC2 c1(C(=O)OC)c(C)cc(C)nc1NC12C(CC(=O)OCC)CC(CC1)C2 C(=O)(CS(=O)(=O)C1CC1)NCc1ccc(CNC(CCC(N)=O)=O)cc1 C(=O)(CS(=O)(=O)CC(F)(F)F)NC1C(CNC(COCCCC#C)=O)C1 N1(C(Cc2nnc(C)o2)=O)CCC(O)(CN(C(=O)C(C)Cn2cccn2)C)C1 CC(=O)CCN=C(NCc1nnc2n1CCCCC2)N1CCC(c2nncs2)C1 C#CC1CN(C(c2cnc(O)n2C)=O)CCN1C(c1ccc(C)c(C)c1)=O C12(CNC(CCC(=O)NC)=O)CC(NC(C3CCCS3(=O)=O)=O)(C1)C(C)O2 c1(C(=O)NC2C3CC(NC(C=Cc4cnc(C)s4)=O)CC32)cn2cnnc2cn1 C(C)(C(=O)NCCC(=O)N(C)C)COCC(CN(C)C)N(C(=O)COCCCC)C C(=O)(C(C)C(F)(F)F)N1CC(OC)C(NC(c2cnsc2C)=O)C1 N1(C(C(CCC)C(=O)OC)=O)CC(NC(=O)C(O)CC(N)=O)CC12CCOCC2 Cc1ccc(CCN(C(=O)COC(C)(C)CNC(=O)CC2CC=CC2)C2CC2)s1 Cc1cc(C(=O)NCCCC2(NC(=O)CN(C)S(N)(=O)=O)CC2)ccc1[N+](=O)[O-] C1(OC)CN(C(c2cncc(OC)c2)=O)CC1NC(C)=O N1(c2ccnc(C(CC)C)n2)CC2CC(NC(c3ccoc3Cl)=O)CC1C2 c1(C(N2CCCC(NC(CC3(C)CCCCC3)=O)CC2)=O)cnc2n1CCCC2 c1(CC)cccc(C(N2CCC(NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)c1N C1(F)(CNC(C=COCC)=O)CCCN(C(c2cnccc2C(F)F)=O)C1 C(=O)(CC(O)C(C)CC)N1CCC(C#C)(C(N2CC(N(C)CC)C2)=O)C1 c1(C(=O)NC(C)CCCNC(c2scnc2C(C)(C)C)=O)ccc(=O)n(O)c1 c1(NS(CC2CC(=O)C2)(=O)=O)nc2c(F)cccc2n1-c1ccccc1 C(c1cccc(CO)c1)=C(CN1CC(C(=O)Nc2ccc(COC)cc2)C1)C#N N1(C(c2nncc(OC)c2)=O)CC(NC(c2ncnc(O)c2F)=O)CC1(C)C C1(NC(c2c(C)nc(Cl)s2)=O)CN(C(c2c(F)cncc2F)=O)CC(F)(F)C1 C1(C(=O)NC(CC2CCOCC2)C(=O)NCCn2cnc(CO)c2)CCC(F)(F)C1 c1(OC)ccc(C(=O)NCCOCCN(C)C(c2cncc(C)c2)=O)c(F)c1Cl N1(C(Cc2c(NCC)cccc2)=O)CCCC2CN(C(=O)CS(=O)(=O)NC)CC12 c1(C(=O)NCC2C(CC(=O)N(C(C3CCOCC3)C)C)C2)nn(C)cc1Cl N1(C(c2cncc(OCC)c2)=O)CCCC12CCN(C(c1ncc[nH]1)=O)C2 C(CC(C(=O)N(CC(C)OC)C)NC(=O)C(c1ccccc1F)C)=CC N1(C(Cn2c(C)ncc2)=O)CCCC(O)(CNC(=O)C(C)S(N)(=O)=O)CC1 CCCC(CC(C)C)C(=O)N1CC(F)CC1C(=O)N(CCC(=O)NC)C N1(C(C(CC)CC)=O)CCCC1C1CCCCN1C(c1cc(C)c[nH]1)=O C1(N(C(=O)NC2CCN(CCOC)C2)CCn2cccn2)CN(C)CCO1 c1(NC(=O)NC2CCC(C)C2)ccc2c(Br)nn(C)c2c1 C1(CCNC(CCCOC)=O)CCCCN1C(=O)C(C)Cn1ccnc1 C1(C2CCN(C(=O)CCc3cccnc3)C2)(NC(=O)CC2NC(=O)NC2=O)CC1 c1(C(N2CCCC(C)(NC(=O)C(O)C(F)F)C2)=O)cc2ccc(F)cc2s1 Cc1csc(Cl)c1C(=O)NCc1cccc(NC(=O)COCCF)c1 N1(C(c2cc(CCC)[nH]n2)=O)C2CCC1C(NC(=O)C(C)CSC(F)(F)F)C2 C(=O)(C1=C(Cl)CCC1)NCC(c1ccccc1)NC(C1C(OC)C1)=O CC(C)CCCC(=O)NC1CCCCC1NC(=O)C(C)Sc1ccc(F)c(F)c1 C(=O)(C(C)(C)C(=O)N1c2ccn(c2)CC1)OC.c1cnn(C)c1.C1C(=O)N1.OCC C1(N(C)C)CCCCC1CNC(=O)CCN(C(=O)CCCn1ccnc1)CCO N1(C(c2c(C)nsc2N)=O)CCC(C)C(NC(=O)CC2CCOC2)C1 C1(OC)CC(c2cn[nH]c2)N(C(=O)CCCN2CCCCC2)C1 N1(S(CC(=O)NCCSCC)(=O)=O)CCNC(=O)C1c1ccc(C)cc1 C1(NC(c2cc(=O)cc[nH]2)=O)CC2C1CCN2C(c1cc(C(F)(F)F)no1)=O c1(C(N2CCC(C(N3CCCC3CO)=O)C2)=O)cc(Br)cc([N+](=O)[O-])c1F C1(NC(CCNC(=O)OCC)=O)COCC1CNC(c1nc(C)no1)=O CC1CCN(C(=O)C(CC2CCOCC2)NC(=O)CCC2CC2)CC1 N1(C(=O)C(c2cccc(F)c2)C2CC2)CCN(C(=O)C(F)(F)C2CC2)CC1CF C1(C(N2CCC(CN(C(c3cc(C)sc3C)=O)C)C2)=O)CCCNS1(=O)=O CCC(O)CCc1cn(C(C)C(=O)N(C(C)C)Cc2ccc(SC)o2)nn1 O=[N+]([O-])c1ccc(Br)c(CNC2(C3CCCCC3)CC2)c1 C(=O)(C(CC)C(C)C)N1CC(CC)C(C(=O)NCc2cnnc(C)c2C)C1 c1(OC)cc(OC)cc(C=CC(N2CCN(C(=O)CC3(C)CC3)CC2CF)=O)c1 C1(C(=O)NCCOC2CCN(C(C=CCC)=O)C2)CCS(=O)(=O)N1 N1(C(c2ccnc(C(C)C)n2)=O)CC(NC(=O)C2=NOCC2)CC2(CC2)C1 N1(C(=O)Nc2ccc(O)cc2O)CCCC2(C1)CN(CC1COCCO1)C2 C1(c2c(C(=O)NCCC3CC=CCC3)nco2)CCCN(CC)C1 Cc1cccc(O)c1C(=O)NCC1CCN(C(C2CCCCC2O)=O)C1 c1(C(=O)NC(C(CO)NC(C2N(CC)CC2)=O)C)cc(C)c(Cl)cc1F C(=O)(CC(C(F)(F)F)NC(C1CCC(=O)N1)=O)NCCc1c(C)nn(C)c1 CC1=C(C(=O)N2CC(CO)(NC(=O)Cc3cccnc3)C2)CCCO1 N1(C(CC(CC)C(C)C)=O)CC2CCCC(C1)N2C(c1ccnc(F)c1)=O c1(CC)cc(S(=O)(=O)NNC(=O)C(N)CO)ccc1OC.OC C1(CNC(CNC(C)=O)=O)CN(C(c2cc(C(F)(F)F)cc(O)c2)=O)CCC1C N1(C(Cc2n[nH]c(=N)s2)=O)CCC(O)(CCNC(=O)Cc2cocn2)C1 N1(C(C(=O)NCC)=O)CCN(C(c2ccnn2C)=O)CC1CCO C1(C)(COC)CCN(C(=NCCOC)NCC2CCCC2c2ccccc2)CC1 c1(CC(=O)N(C(CCNC(CC(C=C)C)=O)C)C)cn2ccsc2n1 C1(NC(=O)C=Cc2cnc[nH]2)CC2(C1)CC2C(=O)NCc1noc(C2CCC2)n1 CCCCCCC(C)C(=O)N(C1CCCN(C(=O)C2=NNC(=O)CC2)C1)CCO c1(NCC(=O)NC(C)(CNC(=O)CCN2CCCC2)C2CC2)ccccc1Cl C1(CNC(C2C(NC(c3cncc(C)n3)=O)CC2)=O)CCCCC1(C)C Cc1cc(C(=O)NC(CNC(C2(CCF)CCC2)=O)C2CCC2)c(O)c(C)c1 N1(C(c2c(C)ccc(C)n2)=O)CC2(C1)CN(C(C1CC(C#N)C1)=O)CCO2 c1(C(N(C)Cc2cc(Cl)on2)=O)cc(O)nn1C C1(O)(C(C)NC(=O)C=CCO)CN(C(c2[nH]ccc2Cc2cnn(C)c2)=O)C1 C(CCCCC(=O)Nc1ccc(F)cc1O)NC(C1CC2(CC2)CO1)=O N1(C(c2c(OC)nsc2)=O)CCCN(C(=O)CC2CCCNC(=O)C2)CCC1 C12(NC(=O)CO)CCOCC1CN(C(c1cc(F)ccc1C(F)F)=O)C2 O=C1CCCC(CC(=O)NC2CCCN(C(=O)C(O)Cc3ccccc3)C2)N1 C(=O)(C(F)(CNC(=O)C(C)N1CCCC1)C(C)C)Nc1ccc(COC)s1 CCC(C)(C(=O)NC1CN(C(c2ccc(Cl)c(C)c2O)=O)CC1C)C(N)=O N1(C(c2n(C)cc(Cl)c2)=O)CCC2(C1)CN(C(=O)CC1CCCC1)CCO2 CCCCCC(O)C(=O)N1CCCCC1C(C)NC(c1cnc(N(C)C)s1)=O Cn1cc(C(O)C(=O)NC2CN(C(C)(C)C)C2Cc2ccccc2)cn1 N1(C(c2c(C)onc2-c2ccccc2)=O)C2CCC1CC(NC(=O)CC(C)O)C2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(=O)C=C3CCC(C)C3)CC2C1 n1(C(C)C)ccc(C(N2CC(NC(=O)CN3CCS(=O)CC3)C(O)C2)=O)cc1=O Cc1c(C(=O)NCCC2CCCN(c3ncnc(=N)[nH]3)C2)cnn1CC(C)(C)O N1(C(C2(CSC)CC2)=O)CC2(C1)CN(C(=O)CCc1ccc(C)o1)CCO2 C1(C(=O)NC(C23COC(CF)(C2)C3)CNC(=O)Cc2cc[nH]n2)CCS(=O)(=O)C1 N1(C(CC(CC)C)=O)CC(C(=O)Nc2ccc(C)c(I)c2)CC(F)C1 C1(C(=O)NCCCC(c2ccccc2)NC(=O)OC(C)(C)C)CC2CCC2C1 C1(CNC(c2c(O)ncc(CC)c2)=O)CC2CCC(C1)N2C(=O)CS(C)(=O)=O C(=O)(C1=CCCCCC1)N(CCC(C)NC(C1C2CC3C(C2)C13)=O)C c1(OC)ncc(F)cc1C(N1CCC(F)(C(=O)Nc2ncc(CO)cc2Br)C1)=O c1(C(N2CC(OC)C(NC(C3C4CNC(=O)C34)=O)C2)=O)cc2cc(Cl)ccc2o1 N1(C(C2C(C(=O)OC)CC2)=O)CCC2(CCN(C(c3csc4nnsc34)=O)C2)C1 c1(C(=O)NC2C(CNC(C(CCSC)NC=O)=O)CC2)onc2cc(C)ccc12 c1(C(N2CC(c3c(NC(C(C)C)=O)nco3)C2)=O)cccc(C2(C)CCO2)c1 C(=O)(C1CCCc2ncnn21)NCCC(C)(C)NC(C(CC)C(C)(F)F)=O C1(C2CCCN(C(C3(C#N)CCCOC3)=O)C2)(NC(C(CC)C(C)C)=O)CC1 O=S(=O)(c1ccc(OC(F)(F)F)c(F)c1)NC(CC(F)(F)F)C(=O)O C(C(C)(C)CC(=O)NCC1(CNC(c2ccc(N)c(N)n2)=O)CCCCC1)OC C1(NC(CCCCC#C)=O)CCN(C(c2cncc(N)c2)=O)CCC1CO c1(CC)ccc(CC)c(NC(=O)C(=O)NC(c2nc(C)no2)C(C)C)c1 C1(C)(C(N(CCN(C(CS(CC)=O)=O)C)C)=O)CCC(C(=O)OC)C1(C)C C1(CN(C(=O)C(C)NC=O)CC)CCN(C(C2CCCOC2C)=O)CC1 CCC(CC)C(C(=O)N1CCS(=O)(=O)C(CCNC(=O)CCOC)C1)OC C1(CN)CCCCN1CCOC.C1(C(=O)OCC)(OC2CCNCC2)CCCC1 c1(OC)cc(C(=O)NC(C(=O)N2CC(NC(C)=O)C2)C2CC2)on1 C(=O)(CCC(=O)NN(C)C)N1CCCC(CC)(NC(=O)C(C2CCC2)OC)C1 N1(C(CCNS(C)(=O)=O)=O)CCCC(CCCCOCCC2CCC(O)C2)CC1 O=C(C1=CC2CCCC12)NCC1CCCN1C(c1nccn2ccnc12)=O N1(C(C2(C)CCCO2)=O)CCCC(NC(C2CCC(O)CC2)=O)CC1 c1(C2(C(=O)NCC(C3CCCC3)NC(C(c3cccnc3)C)=O)CC2)cccnc1 C(N=c1nc2scnc2c(NC2CC2F)[nH]1)c1scc(COC)c1 N1(C(c2cccc(C)n2)C(=O)NCC2CC2)Cc2cncnc2C1 C12(NC(c3cnc(O)c(Cl)c3)=O)CCC1CN(C(=O)C(F)(F)c1ccccn1)C2 C12CC(C1)CCC(=O)N2.N1(C(COCC(=O)OC)=O)CCC1CC1CCCC1 C(c1ccc(Cl)cc1F)=CC(N1C2(CN(C(C34CC(C)C3C4)=O)C2)CC1)=O c1(NC(=O)CC2CCN(Cc3ccncc3O)C2)cccc2scnc12 c1(C(=O)NC(CNC(C2C(COC)C2)=O)(C)C)ccn2cncc2c1 Cc1nc(N2CCCC(C)(CNC(c3cc(CF)on3)=O)C2)cc(C#N)n1 N1(C(C(CC)C#N)=O)CC2(CCCC(CNC(c3ccn4nccc4c3)=O)O2)C1 c1(C(=O)NC2COC3(C2)CN(C(=O)C=CCF)C3)ccc2c(c1)COCC2 c1(C(=O)NC(CC(C)NC(c2n[nH]cc2Cl)=O)C)ncn2c1COCC2 N1(C(C(C=C)O)=O)CCN(CC2(NC(=O)C(=Cc3ccco3)C)CC2)CC1 CC(C)C(O)C(C)C(=O)NCCOCC(=O)NCCC1(O)CCCCC1 N1(C(=O)CCN=c2nc[nH]s2)CCC(CO)C12CCCC2 c1(OC)c(C(=O)NC2(C)CN(C(=O)C(C)C(F)F)C2)ccc2c1CCC2 c1(CC2N(C(C(COCC)n3cc(-c4cc[nH]n4)nn3)=O)CCCC2)cccc(Br)c1 c1(CCC)ccc(C(C(=O)NCCOC)N(CC#N)CCOC)s1 CCCCCCCC(=O)N1CCC(C)(NC(C2CCOC2C2CC2)=O)CC1 CON(CCC(=O)NCCC(C)N(C)C)C(=O)C1CCC2(CCC2)C1 N1(C(CC(C=C)CC)=O)CCOC2(C1)CN(C(=O)C1=NOCC1)C2 Cc1ccc(CC(=O)NCC2COCC2NC(=O)CC2=CCCC2)c(Cl)n1 S(=O)(=O)(c1cccc(N2CCOC(C)(CCO)C2)n1)N1C(C)CCCC1 Cc1c[nH]cc1C(=O)NC1(C(=O)NC2CCC2C)CC1(C)C C1(C)(NC(Cc2ccc(CCC)cc2)=O)CCCN(C(=O)Cc2ccccn2)C1 c1(CC(C2(NC(=O)C=CC(C)C)CC2)NC(C(C2CCC2)OC)=O)ccccc1F c1(C(=O)NCC(CC(=O)OC)(C)O)c2c(nn1C)CCS(=O)(=O)C2 c1(C(=O)NC(CN(C(C(C)NC(C)(C)C)=O)C)C)cc(O)nn1C C1(CNC(c2cn(C)nc2)=O)COCCN1C(c1cnc(O)s1)=O c1(CC)cnc(O)c(C(=O)NCC2(C)CN(CC)CCO2)c1 C(C(F)C(=O)N1CCC(c2nn[nH]n2)C1)C1CN(C(CC2CC(CC)C2)=O)C1 c1(-c2nnc(C(C)(C)C)o2)ccc(Cl)cc1Cl.N1CCOCC1 C1(NC(c2n(CCC)ccc2)=O)CC(C)CN(C(=O)CCC(C)(F)F)C1 CC1(C)CCC(CCNC(=O)NC2CC(CC(F)(F)F)C2)OC1 C(=O)(C1=CC2CCCC12)N1CCN(C(CC2C(C)C2)=O)CC1 N1(C(CNC(CN(c2cnn(C)c2)C)=O)=O)CCSC2CCCC12 C(=O)(C1=C(Cl)CCC(C)C1)NC1(CNC(C2(C(=O)OC)CC2)=O)CCCCC1 N1(C(COC2(C#C)COC2)=O)CC23CCCCC2(C1)CN(C(c1cnn[nH]1)=O)C3 C12(NC(c3c(OC)c(F)ccc3)=O)CCCC1N(C(=O)C(C)S(N)(=O)=O)CCC2 c1(C(C(=O)N(CCN(C(=O)C(F)n2ccnc2)C)C)(C)C)ccc(Br)cc1 C(=O)(C1c2c[nH]nc2CCC1C)NCCCN(C(c1n(COC)ncc1)=O)C1CC1 Cc1cc(Cl)c(CNc2ccc(NC(C3(CN)CC3)=O)c(C)c2)c(Cl)c1 C1(O)(CNC(c2ccn(CC)c2C)=O)CCCN(C(c2ccc(CO)s2)=O)CC1 N1(C(C(C(=O)OCC)CC)=O)CC(NC(C2CC(OC(C)(C)C)C2)=O)C(C)(C)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CC(C2CN(C(=O)C(C)Cc3ccco3)C2)C1 N1(C(COCC(=C)C)=O)CCN(C)C(C(=O)NC2(C)CCCC2(F)F)C1 C1(NC(=O)C(C2CCOCC2)O)CCN(C(=O)NC2CC2c2ccc(Cl)s2)CC1 C1(CCC)CN(C(c2cc(C(N)=O)cn2C)=O)CCN1C(=O)COCC1CC1 C1(C(=O)NCCN2CCCC2)C(C2CC2)CCN1C(=O)CC1CN2CCC1CC2 C1CCCCC(=O)N1c1ccc(O)c(C)c1.C(C)(C(=O)O)NC(C)=O c1(C(N2CC(OCCNC(C3CC3Cl)=O)C2)=O)ncsc1Br c1(C(=O)NC2CC(F)(CNC(CC(CC)O)=O)C2)c(F)cccc1[N+](=O)[O-] O=C(CS(=O)C(F)(F)F)NC1CC(CNC(c2ccc(C3CC3)nc2O)=O)C1 C(=O)(CC(CN(C)C)CC)NC(CC=C)CNC(c1ccc(C(C)C)nc1O)=O C(=O)(CCC(=O)NN(C)C)NC1C(C=C)CN(C(=O)COCC2CCC2)C1 c1(C(=O)NCC(C)(CO)NC(C2CCC(C(N)=O)O2)=O)ccc2c(c1)CCN2 CC(CC(C)(C)C)C(=O)NC(C)(C)CC(=O)N1CC(O)C1 O=C1OCCC2CN(C(C3(NC(=O)CC4CCC(O)C4)CSC3)=O)CC12 c1(C(=O)NCCn2cc(Cn3nccc3C(=O)O)nn2)ccnc2ncnn12 C1(OC)CN(C(=O)C(=O)NCc2cccc(CS(C)(=O)=O)c2)C(C(=O)O)C1OC c1(NC(C2CCCN(C(Cc3ccc(OC)cn3)=O)C2)=O)cc(O)cc(F)c1 Cc1ccc(C(N2CCC(C(C)NC(c3nc(Cl)c(Cl)s3)=O)C2)=O)n2nccc12 c1(-n2c(C(CC(C)SC)N(CCS(N)(=O)=O)C3CCCC3)nnn2)ccccc1C N1(C(CCOC2CN(C(C)=O)C2)=O)CCN(C(C2CC(=O)N(O)C2)=O)CC1 c1(NC(=O)NCC(c2cc(N3CCN(C)CC3)ncc2)(C)C)ccc(Cl)c(Cl)c1 N1(C(C23CCC(C(C)=O)(C2)C3)=O)CCCCC(NC(C2(C)CC(C)=NO2)=O)C1 C1(NC(C(C)N(C)C(c2cc[nH]c(=N)n2)=O)=O)CCC(O)C(O)C1 C1(NC(CCN(C)C(C2(C)CCOC2)=O)=O)CC(=O)N(C2CC2)C1 C(=O)(CCCC(=O)OC)N(C)CCN(c1ccccc1)C(=O)COCCCF Cc1c(F)ccc2[nH]c(C(=O)NC3CN(C(=O)Cc4cc[nH]n4)CC3C)cc12 N1(C(c2c(CC)ncs2)=O)CCC(C)C1CNC(=O)CSCc1cscn1 N1(C(CCC(=O)NCC)=O)CCOC2(C1)CN(Cc1cccc(C(C)(C)C)c1)C2 c1(C(C(=O)NC)N(CCN(C)C)C2CC2)ccc(CC(C)C)s1 Cc1n[nH]c(=NC2CC3CN(C(c4oc5ccccc5c4Cl)=O)CC23)o1 c1(C(C)O)ccccc1C(N1CCC(CNC(=O)CCc2cncn2C)CC1)=O c1(C(=O)NC2CC(NC(C3(CC=C)CC3)=O)CC2O)ccc2cnoc2c1 N1(C(c2c(C)nc(COCC)s2)=O)CCCCC(CNC(=O)C2=COCCO2)C1 C(C(C)(C(=O)NCC(C)O)NCC(=O)NCc1ccccn1)OC CCC(COC)C(=O)NCC1CC(NC(C2(C)CCCCO2)=O)C1 C1(C(N2CC(NC(C(C)SC)=O)C(c3ccnn3C)C2)=O)CC(=O)NC(=O)C1 C1(C(C)(C)NC(c2cnn[nH]2)=O)CCN(C(=O)C(F)C2CCC2)C1 CCCC(C)C(=O)NC1CCCC(CF)C1.c12nnc(S)n1CCNC(=O)CS2 C#CC1(NC(C2(CF)CCN(C(C34CC(C#N)(C3)C4)=O)C2)=O)CCOC1 N1(C(C2N(C(C)C)CCC2)=O)CC2(CCC2NC(=O)CC2CC(=O)NC2=O)C1 C#Cc1c[nH]nc1C(=O)NC(C)(CO)C(=O)N(C1CN(C)C1)C C1(C(=O)NC2(CC)CCN(C(CCC=C)=O)CC2)Cc2ccccc2C1C c1(NC(CC2CN(C(c3ccc(C)nc3)=O)C2)=O)ccc(O)c2ccccc12 N1(c2oc3ccc(C)cc3n2)CCCC2(C=CCO2)CC1 Cc1coc(C(=O)N(C(C)CNC(c2cn(C(C)C)nn2)=O)C)c1C CC1CN(C(C2CCC2)=O)CCC1CNC(=O)COC(F)(F)C(F)(F)F C(=O)(C(F)C(=O)NCCC1CC(C(N2CC(O)(c3nn[nH]n3)C2)=O)C1)OC c1(CNC)c(COC)cccc1F.c1(OC)ccc(C(c2ccccc2Cl)=O)nn1 C1(C#N)(C(=O)NC2CC(C)N(C(=O)CN3CCC(O)CC3)C2)CCOCC1 C1(NC(=O)OC(C)(C)C)CCCCCC1NC(=O)Cc1cc(O)cc(Br)c1 c1(NC(C2CCOC(c3cccc(F)c3)C2)=O)nc(Cl)sc1Cl C1(c2n(C(C)C)nnn2)(NCC2CC3(CC3)C2)COCC1CCF c1(CC(C)C)cc(C(=O)NCCOCCCNC(=O)C(C2CCCCC2)C)on1 CCC(C(=O)NCC1(NC(C2CC2COC)=O)CCC1)c1ccccc1 C1(NC(C(C)(C)NC(=O)NCC)=O)C2CN(C(c3ccc(CSC)[nH]3)=O)CC12.SC c1(C2(OC)CN(C(c3sccc3C3CC3)=O)C2)ccccc1F Cc1c(NC2CCSC(C)C2)ncnc1N(CCCCCO)C C12(C(=O)NCCCNC(=O)NC)CC(CO1)N(C(C1CC3CCCC3C1)=O)C2 C1(NC(Cc2cn(CC)nc2)=O)CS(=O)(=O)CC1NC(=O)CCc1ccco1 C(N=c1nc2scnc2c(NC(c2cccc(Cl)c2Cl)C)[nH]1)c1n(CC)ncc1 CC1NC(=O)OC12CN(C(=O)C=CC1CCCN1C(=O)CC1OCCCO1)C2 Nc1cnnc(NNC(=O)NC2CCCSC2)c1Cl c1(C(=O)NCCC(C)N(CCC)C)cc(CNC(C2CC2(Cl)Cl)=O)on1 N1(C(Cc2c(C)cnn2C)=O)CC2(CC(NC(C3(N=[N+]=[N-])CC3)=O)CO2)C1 C1(NC(=O)Cc2cn(Cc3cccc(Br)c3)nn2)CCCCCC1 C1(C(=O)OC)CN(c2nnc(CCCC3(C)CC3(F)Cl)n2CC(C)C)C1(C)C Cc1cccc(C(=O)NCC2COCCN2C(=O)Cc2cc(F)cc(F)c2)c1Cl C1(C(N(C)Cc2cnc(C)s2)=O)CC2(CCC2)CN1C(C1CCOC1)=O c1(C(N2CC(N(C(CCCC(C)C)=O)C)C(C)(C)C2)=O)cccc2c1CCCC2 c1(NC(C2CC(F)CN2Cc2cncs2)=O)cccc(-n2cccc2)c1 c1(NC(C2(C=C)CCC2)=O)ccc(NC(C2CC2C(C)C)=O)c(C)c1 CS(=O)(=O)C1CC(Cc2cn(CN3CCCC3=O)nn2)C1 N1(C(c2cc(C)c(C)s2)C(=O)NCC(F)F)CCOC2(CCCCC2)C1 C1(C(=O)NC2(CCO)CCSC2)COc2cc(F)ccc2C1 C1(C(N(C)C)=O)CCN(C(c2ccc(CN3CCCC3CC3CC3)o2)=O)CC1 C1(C(=O)NC(C)Cn2cnnc2)(CC)CCCN(C(=O)CC2C=NN(C)C2=O)C1 CC(CN=c1cccc(S(=O)(=O)NCCCSCCO)[nH]1)c1nccs1 c1(N(CC(=O)NCC=C)C)nc(C)cc(=NCC(C)c2ccc(F)cc2)[nH]1 C(CC(C)(C)C)(c1n(CC)nnn1)(C1CCOCC1)NC1C(C)CCC1C c1(C(=O)OC)cccc2c1OCC2CNC(=O)CCc1sccc1Br C1(O)(CCNC(C(CCO)N(C)C)=O)CCCN(C(c2cscc2C#N)=O)C1 CC(=O)C(C)(C)CCC(=O)NC1CN(C(c2ccc(-c3ccco3)s2)=O)CC1C C1(c2n(CCSC)nnn2)(NCc2cccc(Cl)c2Cl)CCCN(CC#N)C1 C=C=CCCC(=O)N1CCCC(CNCC2N(C(=O)OC(C)(C)C)CCC2)C1 c1(CCNC(c2nnnn2C2CC2)C2C(CC)C2)ccc(F)cc1F O=S(=O)(c1ccc(Br)cc1NCCN1CCCC1)N1CCCC(CO)CC1 C(CC1CC1)(C(=O)NCCCN1CCCCC1)N(C)C.C1C(=O)NCCO1 C1(C)(CNC(C2CCN(CC)C2)=O)CCCN1C(c1cnoc1C)=O C1(CNC(COCCC(C)C)=O)(NC(=O)CC2CCCSC2)CC(F)(F)C1 C(=O)(C1CCCc2ncc(C)n21)NC(CNC(C(CCOC)(C)C)=O)C C1(CNC(C(CC)(C)C)=O)CCN(C(=O)CSc2cccc(F)c2)CC1C c1(OC)ccc(NC(c2coc(C(C)NC(C3(F)CCCC3)=O)n2)=O)cn1 Cc1[nH]nc2c1CC(C(=O)NC1CC(C)N(C(=O)CCc3ccccn3)C1)CC2 c1(COC)ncsc1C(=O)NC(C1CCCCC1)C(C)NC(c1cnc(C)s1)=O N1(C(c2c(C)nc(CO)s2)=O)CCC(CO)C(NC(c2nnn(C)c2C)=O)C1 C1(CCC(=O)N(CCCCNC(C(C)C2CC2)=O)C)CCC(=O)NC1 C(=O)(C(C)(C)C(N)=O)NC(CCNC(C(N1CC(C)C1)C)=O)C(C)C c1(-c2cn(CCCN(C(CC(C=C)C)=O)C)nn2)ccc([N+](=O)[O-])cc1 c1(C(CNC(=O)NC2C3CCCCC23)O)cc(F)c(F)c(F)c1 c1(OC)ccccc1CC(C)NC(c1cccc(N2CCC2=O)c1)=O CCCCC(C)(F)C(=O)N1CCC(NC(C2CCC(C)(C)O2)=O)C(F)C1 C(CC(C)(c1nnnn1CC1CCOCC1)NCCNc1scnc1C)SC N1(C(Cc2ccc(SCC)cc2)=O)CC2(CCCCC2NC(C)=O)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NCC1OCCN(C(C2(C(=O)NC)CCC2)=O)C1 N1(C(CC(CC)(C)C)=O)C2CCC1CN(C(c1cccc(OC3CCC3)c1)=O)C2 n1(CCC(=O)NCC2(CNC(C3C(CC)OCC3)=O)CC2)c(C)cc(O)cc1=O N1(C(c2c(CNC(CC3C(=O)NCCC3)=O)ccs2)=O)CCOC2(CCC2)CC1 CN1CCN(C(c2ccc(=O)oc2)=O)C(CNC(c2cc(C(F)F)cn2C)=O)C1 c1(C(N2CCC(CCOC)(NC(CC(=O)NC)=O)C2)=O)ccsc1S(C)(=O)=O C(CCF)(C(=O)NCCC(=O)NOCc1cccnc1)OC c1(N(C)C)nc2cc(NC(=O)CC3CS(=O)(=O)CCN3C)ccc2o1 C(=O)(C1COc2ccccc21)N1CC2CCC(NC(C3CC3(F)F)=O)CC2C1 c1(C(N)=O)ccc(C(=O)N(CCCNC(=O)COC2CCOC2)C2CC2)cc1Cl c1(C(N2CCCC(C)(NC(c3cnc(C)n3C)=O)C2)=O)cccc(S(C)(=O)=O)c1 c1(N(C)Cc2n(CC)cnn2)[nH]c(=NC2CCOCC(C)C2)nc2scnc12 CCCC(C(=O)N1CCCC1C(C)NC(c1cnn(CC(F)F)n1)=O)NC(N)=O CP(C)(=O)C(O)C(=O)NCCN1CCC(NC(=O)CC2CC(F)(F)C2)CC1 c1(C(C)NC(=O)C(C)(F)c2ccccc2)ccc(Cl)cn1 c1(C(=O)NCCCNC(C(c2cccc(F)c2)C)=O)noc2c1CC(C)(C)CC2 C1(C(N2CC(CC)SCC2)=O)CN(C)CCN1C(=O)C(N1CCCCC1)C c1(C(N2CC(CN3CC(CC(C(=O)OC)F)C3)C2)CC)cccn(C)c1=O Cc1cc(C(N2CCCC(CNC(C3(C(F)F)CCC3)=O)CC2)=O)cc(F)c1 c1(OC)ccc(C(=O)NC(C)CCN(C(=O)C(C)CO)C)c(OC)c1 c1(C(NOCCCC=C)=O)cccc(CNC(c2ccncc2CC)=O)n1 N1(C(C2(C(C)(C)O)CC2)=O)CC2CC1(C(N1CCC(OCC(N)=O)C1)=O)C2 c1(C(=O)NCCC2(CNC(CSC)=O)CC2)cnc2c[nH]nc2c1 c1(C(N2C(C)CN(C(C3CC(C)(CC)C3)=O)C(C)C2)=O)cccc(P(C)(C)=O)c1 C1(COC)(NC(C2CCCC(C)(C)O2)=O)CCCN(C(=O)CC(C)(C)C)C1 N1(C(c2cc(OC)ns2)=O)CCC2(NC(=O)C=Cc3cnc[nH]3)CCCC12 N1(C(=O)OC(C)(C)C)CC2CC2(NCc2snnc2C2CC2)C1 c1(C(=O)NCC2C(NC(c3csnn3)=O)C2)ccccc1CO Cn1cc(NC(C2CC(C)(NC(=O)CCSC(F)(F)F)C2)=O)n(C)c1=O C1(C(=O)NCC(C)CN(C)C(c2ccnc3[nH]ncc23)=O)CCCC2(CCC2)C1 CS(=O)(=O)c1cccnc1C(N1CC2CC2(CNC(=O)C2=COCCO2)C1)=O C1(C)(COC)CC(NC(=O)CCC(C)C)CN1C(=O)Cc1nocc1C(C)C N1(C(C(C)Cc2ccccc2F)=O)CC2CCC(C1)N2C(=O)CC1COC(=O)C1 N1(C(c2c(C)csn2)=O)CCCCCC1C(=O)NCc1nncs1 C1(C(N2CC(N(C(C(CC)C#N)=O)C)C2)=O)CS(=O)(=O)CC12CC2 C1(C(N(CCCN(CC(=O)Nc2ccccc2O)C)C)=O)CCCCC12CC2 Cc1ccc(Cl)c(N)c1C(N1CCC(NC(=O)C(C)NC=O)C(O)C1)=O CC(O)C(C)(C)C(=O)NC(C1(O)CCCCC1)C(N1CC2CCC(C1)O2)=O N1(C(Cc2snc(C)n2)=O)CCOC(C)(CNC(c2cn(C(C)C)cn2)=O)C1 N1(C(C(C)CC2CCCC2)=O)C(CC(=O)NC2(C3CCCCO3)CC2)C2CCCC12 C(=O)(C1=COCCC1)NCC(CNC(C1(CO)CCOC1)=O)OC CCCCCCC(C)CC(=O)NC1CCC(O)CN(C(c2ccoc2CC)=O)C1 Cc1nn(C)c(C)c1CC(N1CCSCC1CCNC(c1cncn1C)=O)=O c1(C(=O)NC(C)CN2CCN(C(=O)CC3CC=CC3)CC2)ccn2ccnc2c1 S(=O)(=O)(c1csnc1C(F)(F)F)NCCC(=O)Nc1c(C)cccc1 C(CC1CCCC1)(C(=O)NCCN(C(=O)CCc1cnc(C)s1)C(C)C)OC c1(C(N2CC3(CCC(NC(CCC=C(C)C)=O)C3)C2)=O)ccc2sccc2c1 N1(C(CS(CC)=O)=O)CCCC(C)(NC(c2cnn(C3CC3)c2C2CC2)=O)C1 Cc1cc(F)c(CC(N2CCCC(CNC(=O)C(C)(O)C3CC3)CC2)=O)cc1F Cc1ncc(C(=O)NCC(C)NC(=O)C(c2ccc(F)cc2F)C)cc1N Cc1ccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2(C)C)=O)nc1 C(C(C)(C(=O)NC1CCCCC1)NC(C1CCCO1)=O)SC Cc1ccc(C(=O)NCC23CC2CN(C(c2c[nH]cc(Br)c2=O)=O)C3)c(N)c1 C(=O)(C1Cc2c(Cl)cccc21)NCC1CCCC(NC(CCCCOC)=O)C1 C(=O)(CC(C)(C)CC)N(C(CNC(C(CC)OC)=O)C)C c1(SCC)c(OCC(=O)NCC2(F)CC(NC(=O)CCC=C)C2)cccc1CC N1(c2c(OCCC)cccn2)CCC2(CCCCN(C(C3CCSC3)=O)C2)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCC(C)(C)NC(=O)C(O)C(C)SC c1(C(CNC(c2n(CC)nnn2)c2csc(C)c2)C)ccc(C)cn1 C=CCC(CNC(=O)C(F)F)C(=O)NCC(C)(O)C(C)CC c1(CNC(N)=O)ccc(C(N2CC3CC2C3NC(C2CC2Cl)=O)=O)cc1 CCC(=O)CCC(=O)N(CC(C)C(=O)NCC(C)(O)CC)C C1(CN(C(=O)CC(F)(F)F)C)CN(C(=O)CCP(C)(C)=O)CC1(C)C Cc1cc(C)cc(C=CC(=O)NCCCC(C)NC(C2CC(O)C2)=O)c1 N1(C(c2c(C)nncc2)=O)CCC(NC(=O)Cc2c(C)ncnc2C)C(CO)C1 c1(-c2scc(C(N(C3CCOC3)C)=O)n2)ccc(Oc2ccccc2)cc1 c1(C(N2CC(N(C(c3c(CC)c[nH]c3)=O)C)C2)=O)cc(O)c2ccccc2c1 Cc1c(F)ccc(C(=O)NC2CCC(N(C(=O)CC3OCCO3)C)CC2)c1C CCC(CC)CCCNC(=O)C(Cc1ccco1)NC(c1ccc(CO)o1)=O C1(NC(=O)C(F)=C2CC2)CCC(C(=O)NCC)CC1.C1CCNC(=O)C1.C(=O)(OCC)N c1(OC)ccccc1C(=O)NCC(CO)NC(=O)CC1CCC1C c1(CC)c(C(=O)NC2CC(CNC(=O)CC3CCCC3)C2)[nH]c(C)c1CCO N1(C(CC(CC=C)NC(c2nccs2)=O)=O)C2CCC1CC(CO)C2 c1(C(=O)NC2(C)CC2)cccc(O)c1F.c12ccc(cc1)C(=O)NC2CO.COC Cc1ccc(C=CC(=O)N(CC(C)(C)C#N)C(C)(C)C)s1.C1C(=O)N1 N1(C(C(CC)C(C)C)=O)CCc2nc(CNC(=O)C(C)OCCOC)sc2C1 N1(CC(=O)N(CC(C)(C)CNC(c2cn(CC)cn2)=O)CC)CCS(=O)(=O)CC1 C1(C(N2CCC(C)C(CNC(C3(C(N)=O)CC3)=O)C2)=O)C2CCC(C2)C1(C)C C#Cc1ccc(CNC(C2CC3C=CC2C3)=O)cc1.C12CN(CCO1)C2=O N1(C(CCCOCCC)=O)CCOCC(NC(c2ccc(CO)cc2)=O)C1 C=C(C)C1CN(C(=O)C(C2(O)CN(C(c3cn(C)nc3C)=O)C2)F)CCO1 C1(CNC(=O)NC(C)C)CC(c2ccccc2)(OCCCC(=O)OCC#C)C1 C=CC1(C(=O)N(C2CC2)CC2(O)CCC2)CCN(C(=O)CC2CCCNC2=O)C1 C1(OC)CN(C(c2c(Br)noc2C2CC2)=O)CC1NC(c1ccoc1)=O CN1CC=C(C(=O)NC2CCC(CC(=O)NCC34CCC(CC3)O4)C2)C1 c1(-n2ncc(C(N(CC(C)N(C)C(C3C(C)C3C)=O)C)=O)n2)ccc(F)cc1 O=S(=O)(c1cc(Cl)c(Br)cc1F)N1CCN(Cc2ncc3ccccn23)CC1 c1(NC(C(C2CN(C(COC)=O)C2)O)=O)cnc(N(C)C)nc1 c1(C(=O)NCC23CC(NC(C(C)CC(F)(F)F)=O)(C2)C3)ccc(F)c(Cl)c1N N1(C(C(N2CC(c3ccc(C)s3)OCC2)=O)C)CCc2ccccc21 C(=O)(C(C)(CO)OC)NCC1C(C(N(CC(=C)C)CC)=O)CC1 CCS(=O)CC(=O)N1CCC(C(C)NC(c2cncc(C(C)C)c2)=O)C1 c1(OC)cc(C)ccc1CNC1CCC(C(=O)NC(c2ccc(Cl)cc2)C)OC1 N1(C(c2nn(CC)c(C)c2)=O)CCC(CNC(c2cc(C)c(C)o2)=O)C12CC2 c1(C(=O)NC(CC)CN(C(=O)CCc2csc(=N)[nH]2)C)cn2ccsc2n1 CN1CC(O)CC1C(=O)NCC1CC1CC(=O)NCC(C)(C)C1CCCC1 C(c1ccccc1Cl)=C(C(=O)NC1CCN(C(C2(CC)CCOCC2)=O)CC1)C C1(C)(NC(C2OCC(C)C2)=O)CCCN(c2ccncn2)C1 c1(C(N2CC(C)(NC(=O)CNC(=O)Cc3ccccc3)C2)=O)cncc(N)n1 c1(C(=O)NC2C(NC(=O)C=CC3CC3)C2)c(-n2cccc2)sc2c1CSC2 C(CC(C(=O)NC(CC1CC1)C(=O)NCCCC1CCC1)N(C)C)N(C)C N#Cc1cc2cc(C(=O)NCCNC(c3cnn[nH]3)=O)[nH]c2cn1 c1(OC)cccc(Cn2cc(C(=O)NCC(O)CNC(=O)CC3(C)CC3)nn2)c1 n1(CCc2nc(-c3cncs3)nn2Cc2c(C)cccc2)cnc2ccccc12 C1(C(=O)OC(c2cccnc2)C2CC2)CC2(CCN2C(=O)NCC)C1 N1(C(CN(C(=O)CCC(C)OC)CCC)=O)CCCC2CC1C2(C)C c1(CC)ccc(C(N2CCC(F)(CNC(C3OCCOC3C)=O)CC2)=O)c(F)c1 Cc1ccc(CC(=O)N(C2CCCC2)CCN(C)C)cn1.C12(CCC1)CC(=O)N2 C1(C(N(CC(C)NC(C2CCC(C(F)F)CC2)=O)C)=O)C2CCC1(C)C2(C)C C1(NC(CC(=O)OC)=O)C2CC3C1C3C2C(=O)Nc1cccc(C)c1 c1(SC)ccc(N)cc1C(N1CC2CC(NC(C3(C)CCC(C)(C)C3)=O)C1C2)=O C1(C)(C(N2CCC(C=C)C2)=O)CN(C(c2cccnc2)=O)CC1C C1(C(N(CCCF)C)=O)(NC(=O)C(=O)NCC2CC2)CCC(C)(C)C1 c1(C2(C(=O)NC3CN(C(C=CC(CC)C)=O)CC3F)CC2)ccc(C)cc1F C1(NC(C(CCC)CC)=O)CC2(CCN(C(C3(OCC)CCC3)=O)CC2)C1 N1(C(C(C=C)O)=O)CCOCC12COCCN(C(C1Cc3cccnc3C1)=O)C2 CC(C)CCCCC(=O)NCC1CCCOC1C1CCN(C(=O)CC(C)C(F)F)C1 c1(C(=O)NC2(CNC(C3CC(C#C)(O)C3)=O)CCOCC2)nccc(Cl)c1C N1(C(c2ccc(CNC(C(C(C)C)N(C)C)=O)s2)=O)CCCC2(CCC2)C1 N1(C(CCC(CCCN(C)C)=O)=O)CC2(CCOCC2)CC1CC(=O)NC(C)(C)C c1(CNCC23C(CN(C(CNS(C)(=O)=O)=O)C2)C3)ccc(O)cc1Br C=C(CC)CN=C(NC(C)C)N1CCC(OCc2ccccc2C)C1 C1(CNC(c2ncn(CC)c2)=O)CCCCC1NC(c1csc(C)n1)=O N1(C(C2OCCN(C)C2)=O)CC2CC(F)(F)CCC2(N)C1 CCC(CSC)(c1nnnn1C1CCOC1)NCC=Cc1ccco1 c1(C(=O)NC(CNC(Cn2ncc(C)c2)=O)CO)noc2c1CC(C)(C)CC2 c1(C(=O)NCCC(CNC(C2CN(S(C)(=O)=O)C2)=O)C)c(C2CCC2)cnn1C n1(CC)cc(Cl)c(C(N2CCC(CCNC(=O)Cc3ccccn3)C2)=O)n1 c1(C(N2CCCC(NC(CC3(C)CCC3)=O)C2)=O)ccc2c(c1)COC2(C)C C1(C)(NC(C2CC(C(=O)OC)C2)=O)CCN(C(c2cc(C)c(C(F)(F)F)s2)=O)C1 C(=O)(C1=CCC(NC(c2c(Cl)cnn2C)=O)C1)NC(CC)C1CC1 N1(C(c2cc(OC)n[nH]2)=O)CCCC(CCNC(C2(O)CCSCC2)=O)C1 C1(NC(c2cccc(C(F)(F)F)c2)=O)CCCCC1NC(C1(F)CC2(CC2)C1)=O c1(C(=O)Nc2cccc(Br)c2)cc(C2=CCNCC2)c2cn[nH]c2c1 CC1CCC(CNC(c2noc(COCc3ccccc3)n2)C)CC1 C1(CCNC(CCCNC(C)=O)=O)CCCCN1C(c1ccsc1C#N)=O C1(C(=O)NC2(C)CN(C(=O)CC3(C)OCCO3)C2)CC2CCC1C2 C=CC1CN(C(c2cc(F)ccc2-c2cn[nH]c2)=O)CC1NC(=O)C(C)O c1(C(=O)NCC2CCCCN2C(=O)C=C2CCC2)cc2ncccc2[nH]1 c1(CN2CCN(C(c3cc(C(C)=O)c(O)cc3)=O)CC2)c[nH]c2cccc(O)c12 c1(COC)cc(Br)ccc1N(C(C(=O)NC1(C)CC1)C(C)C1CCCC1)C c1(SC(C(N2C(CNC(Cc3cnc(C)s3)=O)CC2)=O)C)ccc(F)cc1 C=CCC(CNC(C1(CC(=O)OC)CC1)=O)NC(=O)CC(C)n1cccn1 C1(CC(N2CC(C(C)NC(C3CC34CCCC4)=O)C2)=O)NC(=O)NC1=O C1(NC(C2(OC)CC2)=O)CCC(C(=O)N(CCCN=[N+]=[N-])C)C1 C(CCC(O)C(=O)NCc1ccc(CO)cc1)NC(C1(C)CCN(C)C1)=O C(=O)(CC(C)(C)C(F)F)NC(C1CN(C(C2CC3(CC(OC)C3)C2)=O)C1)C C=CC1CN(C(C2CC2(Cl)Cl)=O)CCN1C(=O)Cc1ccc(OC)cc1 c1(C(N2CC(C)N(C(C3C=CC(=O)N=N3)=O)CC2)=O)ccc2nc(CO)[nH]c2c1 C1(CCNC(C2(SC)CC(=O)C2)=O)CN(C(=O)C(C)C(F)(F)F)CCS1(=O)=O N1(C(COC)=O)CCc2ccccc2C(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(N2C(C)CC(CC(=O)NCCCOCCO)C2)=O)ccc2ccoc2c1 C12(C(=O)NC(C3C(C(=O)OC)C3)C)CCN(C(C3CCC3(F)F)=O)CCC1C2 c1(OCCC(N2CCC(C)(NC(C3ON=C(C)C3)=O)C2)=O)cc(C)cc(C)c1 c1(-c2ccc(C(F)(F)F)cc2)csc(=Nc2cccc(Cl)n2)n1CC1CC1Cl CCC(CC1CCCC1)C(=O)NCC(F)CNC(=O)CSc1cnn(C)c1 c1(C(=O)NCC(C)CN(C)C(C2C(C)C2(F)F)=O)cccc2nc(O)n(C)c12 C1(C(=O)NCCN(C)CC2CCCN2CCCO)CC(C#N)(c2ccccc2)C1 C1(NC(CC2CC(C)N(C(c3cnsc3)=O)C2)=O)CCC([N+](=O)[O-])CC1 Cc1cn2c(C(=O)NCC(C)NC(C3CCOC(C)(C)C3)=O)c(Cl)nc2s1 C1(C(N2CC(CNC(C3C(CC)CCO3)=O)C2)=O)CCCCC(F)(F)C1 C1(NC(CN(C(C)C)C)=O)CC2CC(NC(c3nc(Cl)c(=O)[nH]c3N)=O)CC2C1 C1(N(C(C(CC)F)=O)CCO)CCN(C(=O)Cc2ccsc2C)CC1 C1(C(=O)NCCCNC(CC2(C(=O)OCC)CCC2)=O)CCCS(=O)(=O)N1 c1(C(=O)NCCC(C)N(C)C(c2ccc([N+](=O)[O-])[nH]2)=O)c[nH]nc1S(N)(=O)=O Cc1cc(N(C)C(c2ccccc2F)C)ccc1NC(N)=O N1(C(C2(F)CCCN(C(C3CN(C)C(=O)CC3)=O)C2)=O)CCOCC(F)(F)C1 C(=O)(C(CC(C)SC)N1CCN(Cc2nc(CC)no2)CC1)NCCCC CCC(COC)C(=O)N(C1CN(C(=O)CN(C)C(c2cncs2)=O)C1)C NC1CCN(C(=O)Cc2ccc(OCC(F)F)cc2)CC1CO C1(n2c(-c3[nH]c(-c4ccccc4)nc3C)nc(C(C)C3CC3)n2)CCC(F)(F)CC1 c1(OC(C)C)c(C(N2CC(NC(=O)CCCC(F)F)CC(C)C2)=O)cccc1N Cc1sncc1C(=O)NC(C)C(C)NC(c1cnc(S)nc1)=O C1(NC(C(C)O)=O)C=CCN(C(=O)CNC(c2cccc(Cl)c2)=O)C1 N1(C(CC(C)OC)=O)CCN(C(=O)C(=Cc2cccn2C)F)CC1C1CCCC1 N1(C(COC2(C)CCC2)=O)CC(NC(C2CC2c2ccco2)=O)C(O)C1 Cc1cc(C(N2CC3C(CNC(=O)C4=COCCC4)C3C2)=O)cc(N)c1Cl CC1(C)CCOC(C(=O)NC2C(NC(C3(C)CCCCC3)=O)C2(C)C)C1 C1(NC(=O)Cc2cn[nH]c2)CCN(C(c2coc(Cl)c2)=O)CC1F N1(C(c2c(C)ccc(O)c2)=O)CCCC2CN(C(=O)Cn3cnnc3O)CCC12 C=Cc1ccc(C(N2CC(OC)C(NC(=O)Cn3ncccc3=O)C2)=O)cc1 C1(C(=O)NCC(C2CCC2)NC(c2cnn(CC(F)F)n2)=O)CCCCS1(=O)=O c1(N(CC)CC23CCC(CC2)C3)ncnc2c1ncn2CC1CCOCC1(C)C C1(CN(C2CCN(C)C2=O)C)CC(F)(F)CN1.c1(-c2nnn(C)n2)c(Br)ncn1C C(=O)(C1=CCCC1C)NC1CN(C(c2ccc(N(CC(C)C)C)cc2)=O)C1 N1(C(C(CSC)OC)=O)CCCN(C(=O)CC(C)(C)C2CC2)CC1 C(=O)(C1CCCc2nncn21)NCCCCN(C(=O)CCC1CC(C)(C)CO1)C C12(CNC(=O)CSCC3CCCCO3)CC(CN1C(c1ccc(Cl)o1)=O)C2 S(=O)(=O)(c1cc(C(N2CC3CC2CCC3O)=O)n(C)c1)NC(C)C C(=O)(C1SCCc2ccccc21)NCC1C(C)CCN(C(c2coc(Br)c2)=O)C1 C1(C(=O)OCC)(C(C)C)CCCN1C(C1COCC(C)O1)=O.N1(CC)CCN1 C1(CNC(c2n(CC)cc(Cl)c2)=O)CCCC2CN(C(=O)C#CC(C)(C)O)CC12 C#Cc1ccc(C(=O)NCC(CCOC)NC(c2ccc(COC)o2)=O)c(C)c1 c1(-c2c(C(=O)Nc3cncc(C#N)c3)n[nH]c2)ccc2c(c1)C(=O)NCC2 O=C(CCCCCCNC(C1(CF)CC1)=O)NCCc1ccnc(F)c1F CCC(C)CCCC(=O)N1CCCC(F)(CNC(=O)COC(C)C)C1 C12(CC(=O)NCC(C)(C)CONC(c3cnc(S)[nH]3)=O)COC(CF)(C1)C2 c1(C(=O)NC2C(NC(=O)C3=NOCC3)C2)ccc2c(=O)c3ccccc3sc2c1 C1(CN)Cc2occ(C(=O)NCC34CCC(CC3)CC4)c2C1 N1(CCN(C(=O)C=C(Cl)Cl)C)CCN(C(C2(c3cccc(Cl)c3)CC2)=O)CC1 c1(C(N(CCOC)Cc2ccccc2C)=O)coc2c1CNC2 c1(OCC)cc(C=CC(=O)NC2CCCCC2NC(=O)CC2CC2)ccc1O C(C(C(C)C(C)C)NC(=O)CN1CC(=O)NC1=O)NC(c1c(SC)n(C)nc1)=O C1(CNC(C(CCC)(C)O)=O)CC2CCC(C1)N2C(C1CCCCC1O)=O Cc1cccc(CNC(=O)C(C)CN(C)C(c2ncccc2N)=O)n1 c1(OCC)ccc(NC(=O)C(=O)Nc2cnn(C)c2C)cc1F N1(C(C2N(S(C)(=O)=O)CC2)=O)CCC(O)(CNC(C2(CC3CC3)CCCC2)=O)CC1 CCS(=O)(=O)c1cccnc1C(N1CC(NC(=O)CC(C)CN(C)C)C(O)C1)=O N1(C(CCC2(C)CC2)=O)CC2CC(C1)CN(C(=O)C(F)(F)c1cncs1)C2 C(=O)(CC1=CCN(C(=O)C(CCC)OCC)CC1)N1CC(C#C)OCC1 C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(N(C)C(c2cnoc2C2CC2)=O)CCCC1 N1(C(C(C)NC(=O)CCCCC2CC2)=O)CCCC12CCCOC2 C1(C(N(C(C)C(=O)N(CC(O)C2CCC2)C2CC2)C)=O)CCCCNC1=O N1(C(C(C)NC(C)=O)=O)CCC(CN(CC(C)O)C(C2CC2CC(C)(C)C)=O)C(O)C1 C(C(C)(C)C(=O)NCCC1CCCCN1C(=O)CC1(C#N)CC1)OC c1(C2C(C(c3cc(C(F)F)no3)=O)C2)cccc(F)c1 C(=O)(C(=O)CC(C)CC)NC(C(N1CCC(C(C#C)C)CC1)=O)CCF c1(C(N(C(C)CNC(=O)CC2CC3(CCC3)CO2)CC)=O)cnc(OC)c(F)c1 C1(C(=O)NC(c2ccc(Br)c(Cl)c2)(C)C)NC(=O)C2CCC12 CC1(C)CN(C(=O)CC23CCCC2C3)CCC1NC(=O)C=Cc1cncnc1O Nc1c(C(=O)NCC2CCCN2C(=O)Cc2ccsn2)cc(F)cc1[N+](=O)[O-] Cc1ccc(Cl)c(C(=O)NCC2CCC2NC(c2cc(C3CCC3)nn2C)=O)c1 Nc1c(Cl)cc(C(N2CCC3(CC2)CC3CNC(c2cscn2)=O)=O)cc1Cl N1(C(CN2CC(C)(OC)C2)=O)CCC(C(=O)NC2CSC2)CC1(C)C C1(C)(NC(c2ccc(C)n2C)=O)CCCN(C(C2CCCCO2)=O)C1 c1(C(=O)NC2C(NC(C3(C)CCCS3)=O)CCC2)cccc(NC(=O)C2CC2)c1 N1(C(C2(C#N)CCCCCC2)=O)CCC(C2(NC(C3CCC4CC34)=O)CC2)CC1 C1(NC(c2c(C(C)(C)C)ncs2)=O)CC2CCC1N2C(C1(C(F)(F)F)CCC1)=O CC1(C(F)F)CCCN(N(Cc2cccc(Br)n2)C2CC2)C1 CCC(CNC(c1cc(C2CC2)no1)=O)(CC)C(=O)N1CCC(C)(C)CC1 Cc1cc(N)c(C(=O)NCCc2ocnc2CNC(=O)CCc2nccs2)cc1C C1(C)(C(C)C)CN(C(C2CC(C)(C)C2)=O)CCO1.C123CC(C1)(C2)CNC3=O c1(C(N2CCCC3(CC(NC(C(N)=O)=O)C3)C2)=O)cc2n(n1)CCCCC2=O C1(C(=O)NC(C)Cc2ccncc2)CC=CCN1C(c1scnc1Cl)=O N1(C(c2n(CCOC)c3c(c2)cccc3)=O)CCc2cc(Br)ccc2C1C(F)F c1(CNC(C(C)OCC2CC2)=O)cccc2c1CCN(C(c1sccc1F)=O)C2 C1(O)(C(C)NC(C(C)OCCCC)=O)CCN(C(=O)C(C)=C2CCC2)CC1 c1(CN(C(C2(C)CC2)C)CC2CC2)cn(CCCO)nn1 N1(CC)C(=O)CCC1C(=O)NCC(C1CCCN1C(c1cccnc1C)=O)(C)C N1(C(COCCC)=O)CCCC1CN(C(=O)CC1CC(F)C1)C c1(SC)cc(C(=O)N(CCCCNC(c2[nH]cnc2C#N)=O)C)oc1C C(=O)(C(C)CC(=O)N1CC(N2CCN(C3(C(=O)SC)CCC3)CC2)C1)OC c1(C(N2C3C(NC(COC4C(C)CCCC4)=O)C(C3)C2)=O)cn2cccnc2n1 CC1CCN(C(C2CN(C(C34CC3CNC4=O)=O)CC2(C)C)=O)CC12CCC2 C1(C)(NC(c2cc(CNC(c3c(C)cn(C)c3)=O)sc2)=O)CC(C)(C)OC1=O c1(SC(C)C(=O)NCCOC2CN(C(C3CCC(C)(C)O3)=O)C2)ccc(F)cc1 c1(OC)ccnc(F)c1C(=O)NCC1(CNC(C2CC(C)OC2=O)=O)CCCC1 C(CC(=O)NCC(C)(O)C1CCCC1)N(C)C(C1CC1(C)C(N)=O)=O c1(C(C)C)ccc(C(N2CC(NC(C3(C4CCCO4)CC3)=O)C(C)C2)=O)c(O)n1 C(CC(CNC(c1snnc1C(C)C)=O)NC(=O)CCc1cscn1)OC CC1CCC2(CO1)CN(C(C1(CNC(=O)CC3CCCC3)CC=CC1)=O)C2 N1(C(C)C)CCC2(CCN(C)C2=O)C1.c12ccc(cc1)CN2C(C)(C)C c1(C(=O)NC2C(CNC(C(CC=C)OC)=O)C2)c(Cl)ccc(OC)c1N Cc1ccc(OCCC(=O)NC(C)(C)CCN(C(=O)C(C)CC2CC2)CC)cc1 N1(C(c2onc(C)c2C)=O)CCc2sccc2C1CNC(C1CCC(O)CC1)=O c1(C(=O)NCC2CCN(C(c3ccc(OC)s3)=O)C2)cc2c(Cl)cncc2s1 Cc1cc(C(=O)NC(CNC(=O)C=Cc2nc(C)cs2)C(C)C(C)C)c(C)cn1 c1(C(N2C3C(CNC(C(=O)N(C)C)=O)C(CCC3)C2)=O)cnc2ccnn2c1 C1(NC(C2(C(C)(F)F)CC2)=O)COCC1NC(c1cc(-c2ccccc2)[nH]n1)=O c1(C(=O)NC2CCCN(C(C(CC)CC)=O)CC2)ccccc1S(C)=O C1(N(C(c2c(C(C)=O)cccc2)=O)C)CN(C(=O)CCCC(C)=O)CCC1C Cc1ncc(Br)cc1C(=O)NCC1CC1NC(=O)Cc1ccc(CO)o1 C(=O)(CC(C)CNC(C1CCCN(C(c2cccc(F)c2)=O)C1)=O)OC c1(CC)nc(C)[nH]c1C(=O)NC(C)(C)CNC(=O)CN1CCS(=O)CC1 Cc1cncc(C(=O)N(C)CCN(C)C(c2cn(CC(F)F)nc2C)=O)c1 c1(C(=O)NC23CC(NC(C4(SCC)CC4)=O)(C2)C3)nnn2c1CCCC2 c1(C(=O)NCC(C)(C)OCC(=O)NCC2(F)CC=CCC2)cccc2occc12 CC(C(O)C(F)F)NC(=O)CCOC1CN(C(C2(C)COC(=O)N2)=O)C1 C1(N(C(C(C)NC(=O)NC)=O)C)CCN(C(=O)CN(C)C)CC1 CCCCN(CCCN(C)C(=O)NC1(CC(C)C)CC1)CC CC1(c2cn(Cc3cnco3)nn2)CCN(C(C2COCCOC2)=O)CC1 c1(CC)cccc(OCC(=O)NCC2(NC(c3ccccc3C)=O)CCC2)c1 C1(F)(C(=O)NCCC(C=C)C)CCN(C(=O)CN(C)C(=O)C2CC2)C1 Nc1c(Cl)cc(C(N2CCC(Oc3cc(Cl)ccn3)CC2)=O)cc1Cl C(=O)(CC1OCc2ccccc21)N1CCC(NC(c2n(C)ncn2)=O)C(F)C1 C1(F)(CNC(C(C2CC2)OC)=O)CCCN(C(=O)CC2CCC(C)O2)C1 c1(C(C)C(=O)N(C(C)CCNC(C2C=CCCC2)=O)C)ccccc1F c1(C2(C(N3CC(NC(C4(C)CC=CCC4)=O)C(O)C3)=O)CC2)ccc(F)c(F)c1 CCC(C)C(C(=O)NCc1cc[nH]c1C(N1CCCCC1CC(N)=O)=O)N(C)C C(C(CC(C)C)C(=O)N1CCOC(C(C)C)C1)NC(c1cccc(C)c1N)=O c1(C(=O)NC2CN(C(c3cc(C)nnc3)=O)CC23CC3)c(F)cc(Cl)cc1F CC1OCCC1CC(=O)NCC(C)(C)CC1CN(C(c2nnnn2CC2CC2)=O)C1 c1(CCCC(=O)NCCCN(C(C(C2CCC2)OC)=O)C)ccc(F)cc1 N1(C(c2coc(Br)n2)C(=O)NCc2cccc(OC)c2)CC2OC(=O)OC2C1 c1(N(C(C2CCN(c3c(OC)c(C)ncn3)C2)=O)C)c(Cl)cccc1[N+](=O)[O-] CCCCC(CNC(c1cc(Cl)ns1)=O)NC(=O)CNC(=O)CN(C)C c1(C(N2C(CN(C(c3c[nH]c(=O)cn3)=O)CC)CCC2)=O)cn(C)c(=O)cc1C CC(C)C(F)C(=O)NC1CCC1CNC(c1coc(Cn2cccn2)n1)=O C1(C(=O)NC(CNC(COc2c(C)occc2=O)=O)C2CC2)CCc2nccn2C1 c1(CCC(=O)N(C(C)CNC(c2cnc(O)n2CC)=O)CC)cn(C)nc1C Cn1nc2cccc(C(=O)NC34CC(NC(c5ccc(=N)[nH]n5)=O)(C3)C4)c2n1 C1(C(=O)NC(CCC)CC)(CC)CCCN1C(=O)CCOCC(F)F c1(OC)cc(=NC(=O)C2(CNC(c3cc(O)nn3C)=O)CCCO2)[nH]n1C c1(C(=O)NCC(CNC(=O)C=CC2CCOCC2)O)c(Cl)ccc2ccoc12 c1(C(C)=O)ccccc1C(=O)NCCC(O)CNC(c1cc(Cl)ccn1)=O N1(C(CSCC=C)=O)CCC(CN(C)C(c2cnoc2CC(C)C)=O)CC1 C(C(=O)N(CCC(=O)NCC1(CC)CCCCO1)C(C)C)(C(C)C)SCC CC1(CNC(C2C=CCN2C(c2cnncc2O)=O)=O)CCOCC1 CC1(C)CCOC1CC(=O)NC1CCCCC1c1ccccc1 Cc1nn2cc(C(N3CCCC(C)(C)C3CNC(C3(O)COC3)=O)=O)nc2s1 C(=O)(C(C)(C)CC1CC1)NC1CCC(CCC(=O)N(CCN(C)C)C)C1 c1(CN(C(=O)CCCNC(=O)C(C)NC(C)=O)CCC)ccc(C)c(Cl)c1 C1(C2(O)CN(C(C3CC=CC3)=O)C2)(CNC(Cc2c(C)cco2)=O)CC1 Cc1c[nH]nc1CNC(=O)C(F)C1CC(NC(C2CS(=O)C2)=O)C1 Cc1cc(C(=O)NC(C)C(=O)NCC(C)NCc2cc(Cl)ccc2F)cc(C)c1 C(=O)(CC(C)(C)C(F)F)NCC1N(C(C(C(C)C)n2ccc(C)c2)=O)CC1 C1(CC)CCC(C)CN1C(C12CC1CCN2C(c1ccnnc1C)=O)=O CCN(OC)C(=O)C1CCCC1CNC(c1n[nH]c(C)c1Cl)=O c1(C(=O)NC2CC(C)CN(C(c3c[nH]nc3C(F)F)=O)C2)cc2cnccc2[nH]1 c1(OCC(=O)NCC(n2cc(CC(C=C)O)nn2)C)ccc(F)cc1 c1(C(N(C2CCC(NC(=O)CCN3CCCC3=O)C2)C)=O)cnc2[nH]ccc2n1 c1(C(=O)NC2COCCN(C(c3ccc(C#C)cc3)=O)C2)cc2sccc2n1C CC1OC2(C(=O)NCc3ccc(CN(C)C(C4CCCC4)=O)cc3)CCC1CC2 CC(C)CC(CNC(C1(C)CC2(CCC2)C1)=O)C(=O)NCCCCC(C)C c1(NC(c2ccccc2Cl)C)[nH]c(=NCC(C)CN2CCOCC2)nc2sccc12 N1(C(C(=O)NCC2(S(C)(=O)=O)CC2)=O)CCS(=O)(=O)CC1.O=C(CC1(CO)CC1)OC c1(NCC(CNC(C2CCCC3C2C3(F)F)=O)O)nccn2nnnc12 CCS(=O)(=O)c1ccccc1C(=O)NC(C1CN(C(C2CC3(CSC3)C2)=O)C1)C c1(CCCCC)nc(-c2cn(Cc3ccccc3)cn2)n(C2CS(=O)(=O)C2)n1 C1(NC(=O)CC2CC2)CCC(C(=O)Nc2c[nH]nc2C(N)=O)OC1 N1(C(CCCOCC)=O)CCC(C)(C)C1CNC(c1cc(C2CCC2)[nH]n1)=O C1(C(N(C(C(=O)OCC)C)C)=O)C=CCCN1C(c1ccc(=N)[nH]n1)=O C1(CC(=O)NC(c2cnc[nH]2)C)CCN(C(c2cccc(O)c2)=O)C1(C)C CC(C)CS(=O)(=O)CCC(=O)NC1CC(CNC(c2cnc3occc3c2)=O)C1 Cc1cncc(-c2cn(CC3CCCN(C(C4CC(F)C4)=O)C3)nn2)c1 C1(NC(CC2CC(OC)C2)=O)CCN(C(c2ccoc2C(C)C)=O)C(C)C1 CC1C(C(=O)NCCCC2CCC2)CCN1C(=O)CCc1ncccn1 C1(=C(CNC(C=CCN(C(=O)C(O)P(C)(C)=O)C)=O)F)CN2CCC1CC2 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCN(C(C2CC3(CC3)C2)=O)C2C1C2 C1(CCNC(C(=Cc2cn[nH]c2)C)=O)CCCCN1C(=O)CCCC1CCC1 N1(C(C(CNC(c2cnc(OC)s2)=O)C)=O)CCCC2(C=CCO2)C1 c1(NC(C(c2ccc(C(C)(C)C)cc2)N(CC(F)Cl)C)=O)ccc(F)cc1F C1(CC)CN(C(=O)Cc2cscn2)CCN1C(c1c(C2CC2)cnn1C)=O CC1(C)CCCCC1=CC(=O)NC1CN(C(=O)CCc2cccs2)CC1O c1(C(=O)NCC2(CNC(C(CC)OC)=O)CCCC2)c[nH]c2nccc-2c1 c1(C(N(C2CC(C(C)=O)NC2)C(=O)CC2(C)COCCO2)=O)ccc(Br)c(F)c1 C1(CNC(=O)OC(C)(C)C)C2CN(C(=O)NC3(Cl)CC3(F)F)CC12 S(=O)(=O)(c1csc(C(=O)NCC2CCN2C(c2ccc(F)cc2N)=O)c1)NC C(=O)(C1CCCc2ccccc21)NC(c1ccc(F)cc1)CNC(=O)C=C(Cl)Cl N1(C(CCC2CCC(C)O2)=O)CCC(CNC(=O)C=C2CCCCC2)CC1 c1(OCC)ccc(CCCC(=O)NCCCNC(c2ocnc2C2CC2)=O)cc1 c1(-c2ncc(C(=O)NCCc3cccc(F)c3)nc2)cnc2cc[nH]c2c1 N1(C(c2ccncc2O)=O)CC(C2CN(C(C3CC3C3CCC3)=O)C2)C1 N1(C(C2C(C)CCC2)=O)CCC(C)(NC(=O)COCCO)C1 N1(C(c2cc(Cl)ccn2)=O)CC2(C1)CN(C(C13CCC(F)(CC1)CC3)=O)CCO2 N1(C(CCc2ccc(C)nc2)=O)CC2CCC2(CC(=O)NCCCCN(C)C)C1 c1(COCC(=O)NC2CCC(CNC(C3C=C(C)CS3)=O)C2)cccc(Cl)c1 c1(C(N2CCC(CNC(=O)C(F)C(F)(F)F)C2)=O)nnn2c1CCCCC2 c1(C(=O)NC(CN(C(c2n(CC)ccn2)=O)C)C)ccc2c(c1)COCCN2 Cn1cnc(CCNC(=O)C(c2cn(C)nn2)NC(c2cnc(O)o2)=O)n1 CC(C)CCC(=O)N(C(CNC(c1ccnc(-c2ccccc2)c1)=O)C1CC1)C CCC(C)(F)C(=O)N1CCC(F)(CNC(=O)CCn2ccnc2C(C)C)C1 c1(Cc2sc(C(N3CC4C(NC(C)=O)C4C3)=O)c(C)n2)nnn2c1CCCC2 C1(NC(Cc2nc(C)sc2)=O)C(C)CN(C(=O)CCCOCCN(C)C)CC1C c1(C(N(C(C)C(=O)NCCC)CCC)=O)cnn(CCOC)c1.C1(CC)(CC)CCC1 CC1CCN(C(c2csc(Cl)c2)=O)CC1NC(C1(C(F)F)CCCC1)=O c1(C(N2CC3(C(C(=O)NCCC(C)N(CCC)C)C3)C2)=O)cc(C#N)cn1C C1(CNC(=O)C=CBr)COC(CNC(=O)CN(c2ncccn2)c2cnccn2)C1 CCCCC(CC)(c1ccccc1)NCC(N1CCC(O)(C(=O)NC)C1)=O c1(C(N2CC(N(CC(C)C)C)C2)=O)ccc(CNC(=O)CC2(C)OCCO2)s1 C1(CNC(C(CC)CC)=O)CCN(C(=O)CSc2ccc(O)cc2)C12CC2 C(C(N=c1nc(C2CC2)[nH]s1)C1CCC1)NC(c1ccn2ncnc2c1)=O c1(CC(=O)N(CC)CC2CCCN2C(c2ccc(C(C)=O)[nH]2)=O)ccccc1C C1(C)(C(=O)NCCC2CC(NC(C3N(CC)CC3)=O)C2)CCN(C)C1 Cc1c(Br)noc1C(=O)NCC1CCCN1C(C1CC1c1ccccn1)=O CC12CCOC(C(N3CC(CNC(=O)C=Cc4ccccn4)C3)=O)(C1)C2 c1(CC(=O)NCCCCc2onc(CC(=O)NC)n2)cnn2cc(F)cc(F)c12 C#CC1(C(N2CC(CCO)(CC)C2)=O)CN(C(=O)C(C)CC)C1 O=C1COCCN1Cc1cccc(C(=O)NCCO)c1.C12(O)CC(C1)C2 C(c1c(C)coc1C)=CC(=O)NC(CCOC)CNC(c1c[nH]c(C(N)=O)c1)=O c1(Cc2onc(-c3cccc(OCC)c3C(F)(F)F)n2)cnc2n1CCCC2 C(=O)(C#CC1(CC)CC1)NC1CC(NC(c2ccc(COC)cc2)=O)C12CCC2 C1(CNC(c2nn(C)c(Cl)c2Cl)=O)CN(C(C2CCCN2C=O)=O)CC(C)(C)C1 N1(C(C23CC(CC)(C2)C3)=O)CCC(C(C(C)C)NC(c2n[nH]cc2Br)=O)CC1 N1(CC)CCCC1C(=O)NC1CCN(C(c2sccc2C(=O)NC2CC2)=O)C1 N1(C(c2cccc(C(C)=O)c2)=O)CCCC2CN(C(=O)CC=C(Cl)Cl)CCC12 C12(CNC(CC=C)=O)CC(NC(C3CCC3C)=O)(CO1)C2 O=C(C1=NOC2(CCN(Cc3cc(O)ccc3Br)C2)C1)NCc1ccc(F)nc1 Nc1nccnc1C(=O)NCC(CO)NC(c1ccc(C(=O)CF)s1)=O CC1(NC(=O)COC2CC2)CCN(C(c2cccc(OC(F)F)c2)=O)C1 c1(C(N2CC(NC(Cc3cc(C)[nH]n3)=O)C3C2C3)=O)cnc2cc[nH]c2c1 N1(C(C(=O)NCC)CCSC)CC(OC(C)(C)C)CC(O)C1 N1(C(C=CC(=O)NCC)=O)CC(OC)CC1(C)CNC(=O)CCOCC C12(C(N3CC4CCC(N(CCCOCC)C)(C3)C4)=O)C3CCC(CC13)C2(F)F Cc1cc(-c2cn(CC(C3CCN(C4CCC4C(=O)O)CC3)F)nn2)ccn1 C#Cc1cccc(C(C(=O)NCC(=C)C)N(C2CCCN(CCC)C2)C)c1F c1(SC2CCC2O)ccccc1CNC(N1CCCC(c2cn[nH]c2)C1)=O C(=O)(C1Cc2ccccc21)N1CCC(CNC(C(C)CF)=O)C12CCC2 C1(C(=O)NC2CN(C(c3cc(C)ncn3)=O)CC(C)C2)CCc2nccn2C1 Cc1c(C(=O)NC2(C(C)NC(=O)Cc3cnn(C(C)C)c3)CC2)nnn1C(C)C Cc1cc(CC(=O)NCC2CC2C(=O)NCC=Cc2ccccc2)ccc1F C(=O)(C(F)C(=O)NCC1(NC(C2(CC(C)C)CC2)=O)CC1)OCC Cc1cc(OCCC(=O)NCC2COCC2NC(C2CS(=O)C2)=O)c(C)c(C)c1 c1(OC)cc(-c2cn(CCCC(N3CCCN(C)C(C)C3)=O)nn2)cc(Br)c1O C1(C(=O)Nc2cc(OC)cc(Cl)c2)CC(N=c2ccn3ncc(C#N)c3[nH]2)C1 C1(CCC)CN(C(C2CCC(C#N)C2)=O)CC1NC(=O)CCOCCCOC Cc1cc2cccc(C(N3CCOCC3CC3CCC3)=O)c2o1 c12ncnc(c1C)NCCCN2C.C(CC(O)C(=O)N1CCCC1)SC C(=O)(C1=CC2C=CC1C2)N1CCC(CC(N2CCC(OC)C2)=O)C1(C)C c1(C(N(CC)CC2N(C(C34CCCN(CC3)C4)=O)CCC2)=O)nccc2ccsc12 C1(CNC(C2(C=C)CC2)=O)C(C)CCN1C(c1c(OC)nsc1OC)=O C1(C(N(S(C)(=O)=O)C2COC2)=O)CC(=O)N(C2CCCCCC2)C1 N1(C(CC2CN(C(c3c(C)n[nH]c3)=O)CC2C)=O)CCCCCC1C C1(NC(C2(CC=C)CCOCC2)=O)CN(C(C2SCCCS2)=O)CC2(CCC2)C1 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC1C(=O)Nc1ccsc1C(C)C C(N=c1[nH]cc2ccnc-2[nH]1)C1CC(NC(C(C)(C)c2sccc2Cl)=O)C1 C=C(CNC(N1CCN(C(n2cncn2)C)CC1)=O)c1ccccc1 N1(C(C(COC)(C)C)=O)CCC(C)C(NC(=O)C(N2CCCCC2=O)C)C1 C1(CNC(C(CC)C2CCOC2)=O)CC(F)(F)CN1C(c1cc(F)ccc1Cl)=O c1(CCC(=O)NCC(c2coc(-c3ccccc3F)n2)(C)C)nnc2n1CCNC2 c1(OC)ccc(C(=O)NCCC2CCN(C(=O)C(C)OCCN(C)C)C2)c(Cl)c1 c1(CN2CC(C(=O)Nc3c(C(C)C)cnn3C)C2)ccc2c(c1)OCCN2C c1(CNC(=O)Cn2cc(Cn3nccc3C(=O)O)nn2)ncnn1C.CCOC c1(CC(C)C)ccccc1CC(=O)NCC(C)Cc1ccc(C(F)(F)F)nc1 CCC(C)CC(C(=O)NCC1(F)CN(C)C1)NC(C1CC(=O)N(CC)C1)=O c1(C(=O)NC2CCN(C(C3(C(F)(F)F)CC3)=O)C2)ccc2c(c1)C(=O)CC2 c1(CNC(NCC(C)S(C)(=O)=O)=NCC2CC(N(C)C)C2)ncnc2c1OCCO2 C1(NC(=O)Cc2cn3ccsc3n2)C2CCC1N(C(C1CCC(F)(F)C1)=O)C2 c1(C(=O)O)ccc(S(=O)(=O)N2CCCC(C(N3CCOC(CCO)C3)=O)C2)s1 c1(C(=O)NC2CC(CNC(c3cc(C)[nH]c3C)=O)C2)ccc(F)c(S(C)(=O)=O)c1 c1(C(=O)NCC(c2ccsc2)NC(C(C2CC2)OC)=O)c(C)cc(Cl)cc1N c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC23CC3)cnn2c1OCCC2 c1(C(N2CC(NC(=O)C(c3cccc(F)c3)O)C2)=O)ccc(O)c(F)c1F C1(CNC(COC2CN(C(C)=O)C2)=O)(CNC(C2CC2[N+](=O)[O-])=O)CCCCC1 C1(C(N(CCNC(c2c(N)sc(C)c2C)=O)CC2CC2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NCC2(C(C)(C)O)CN(C(C(CC)(F)F)=O)C2)CC2(CCC2OC)C1 N1(C(C2CCCS2(=O)=O)=O)CCN(C(c2ccc(O)nn2)=O)C2CCCC12 CN1CCCCC1C(=O)N(CCC1CC1)Cc1cn(CC(=O)O)nn1 c1(NC(CNC(c2cnc(C(=O)OCC)s2)=O)(C)C(C)C)ccc(C#N)cc1F Cn1ncc2c(CN3CCSCC3C(=O)NCc3cnc[nH]3)cccc12 C1(CCC)CN(C(=O)CCn2cccc2)CCN1C(c1ccc(Cl)c(Cl)c1)=O CCN=c1ccc(C(=O)NC2CCC2NC(c2ccsc2C(F)(F)F)=O)c[nH]1 C1(C(N(C2(c3cn(-c4ccncc4Cl)nn3)CCC2)C)=O)CCCN1C=O CC1CC2CN(C(c3ccc(C(F)(F)F)s3)=O)CC2N1C(=O)CC1CC1 c1(C(=O)NC2C=CC(CNC(C3C(C#N)C3)=O)C2)csc2c1CCCC2 N1(Cc2cccc(C)c2F)CCOC2(CCS(=O)(=O)C2)C1 N1(C(C(=O)NCC2C(C)(C)C(=O)C2)=O)CC(C(N2CCOCC2)=O)C(F)(F)C1 c1(NC(c2cc(CNC(C(OCC)OCC)=O)no2)=O)cc2sccc2[nH]1 CC(CF)CC(=O)NC1CCCCC1NC(C1(Oc2ccc(F)nc2)CC1)=O CC1CCS(=O)(=O)CCN1C(=O)NCCc1ccc2ccccc2c1 C12(C(=O)NCC#CCNC(c3cccc(OC(C)(C)C)c3)=O)CCC(C)(C1)OC2 c1(CNC(N)=O)ccc(C(=O)NC2CCCCN(C(=O)C(O)CF)C2)cc1 CCC(CC)CC(=O)NC1CCCCC1C(=O)NCCN1CCCC(O)C1 N1(C(CC2CCC(C)CO2)=O)CCC(C(=O)N(CC(N)=O)C2CCC2)C1CC(C)C c1(C(N2C3(CNC(CN(C(C)C)C)=O)CCC2CC3)=O)cccc2c1CCOC2 Cc1nc(NC(=O)NCC2CCC(=O)NC2)sc1F C1(COCC)C2CCCC1N(Cc1cc(C)cc(F)c1)C2 CC1(O)CCN(C(C2C3CCCC23)C(=O)NCCC2CC2)CC1O CC1CC(C(C)OC(=O)CCNc2cccc(C(C)(C)C)c2)CC(C)O1 c1(C(N2C(CNC(C(C)C)=O)CC(F)C2)=O)cccc(S(C)(=O)=O)c1F C1(NCCSC(C2CC2COCc2cccnc2)C)CN(C(=O)OC(C)(C)C)CCO1 N1(C(C2N(C(C)=O)CCC2)=O)CCCC1(C)CNC(=O)C(F)(F)c1ccccn1 CC1(C)CCCC(C(=O)NCC23CC2CN(C(=O)Cc2coc(C4CC4)n2)C3)C1 c1(CCNC(CCc2cc(C)no2)=O)cc(F)ccc1C N1(C(CCc2cc(C)[nH]n2)=O)CC2(C=C(C(=O)N3CCOCC(C)C3)CO2)C1 N1(C(C(C)=CC)=O)CCCC(CCC(F)(F)F)(NC(c2ccc(SC)cc2)=O)C1 c1(C(=O)NCCNC(c2cc(C(C)C)nc(O)c2)=O)nccn2cnnc12 c1(-c2ccc(C3CCN(c4c(OC)ccc(Cl)c4)CC3)o2)c(F)cccc1F c1(OC)ccnc(C(=O)NC2CN(C(c3ccc(C)n3C)=O)CC2C(F)F)c1F CCCCC(C(=O)OC)N1CC(NC(C2CCN(C3CC3)C2=O)=O)C1 C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(c2c(C)cnnc2)=O)C(C)(C)C1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NC12C(CN(C(COCCC(C)C)=O)C1)C2 C(=O)(C(C#N)C(C)(C)C)N1C(C(=O)NCCC(C)C)CSCC1 C1(C)(C(=O)NC(C)CNC(=O)CS(=O)(=O)N(C)C)CCCS1(=O)=O Cc1nnccc1C(=O)NC(Cc1cnc[nH]1)C(=O)N(C)CCN(C)CCO C(=O)(C(C)C(O)C(C)C)NCCn1ccc(C(NOCCCOC)=O)c1 C(=O)(CCCC(C)C)NCc1nc(C(N(CC=C)CCC)=O)sc1 c1(-c2scc(NC(N3CC(O)(C(C(=O)OC)F)C3)=O)n2)ccc(Cl)cc1 c1(OC)ccc2c(c1)CCC(C(=O)NCCN(C(c1cccs1)=O)C(C)C)C2 Cc1nc(COC2CCCC2)cc(=NCCNCC(c2ccc(F)cc2F)O)[nH]1 C1(NC(C(c2ccncc2)C)=O)CN(S(=O)(=O)C(C)Cl)CCC1(F)F c1(C(=O)NCc2c(C)ccs2)c(Cl)ccc(Cl)c1CO N1(CC(=O)NC2CCC(N(C)C(C3CCNC3=O)=O)CC2)CCCNS1(=O)=O Cc1ccc(NC(=O)C(C)(CO)NC(=O)C(F)C2CCC2)c(C)c1 C1(NC(c2scc(C)c2)=O)CC12CC(NC(=O)CC1C=NN(C)C1=O)C2 C(=O)(C1=CC2CC=CCC12)NCCN(C(c1cc(C(N)=O)cs1)=O)CC c1(NC(C=C(C)CNC(=O)C=CCN2CCC2)=O)ccc(O)nc1 c1(C(N2CCC(NC(C3CC34CC(F)(F)C4)=O)C2)=O)cc2c(cn1)CCCC2 N1(C(c2ccc(C(C)C)cc2)=O)CCCC2C1CCN2C(=O)C=C1CCSCC1 N1(C(C2(CC)CN(C(=O)CC3CCCOC3)C2)=O)CC2CC2C2CC12 C#Cc1ccc(C(=O)NC(c2nocc2C(=O)NCCC(C)(C)F)C)cc1C N1(C(C(C)SC)=O)CCCC2(CCCCC2NC(c2cn(C3CCC3)nn2)=O)C1 C(CNC(C1CC2(CCC2O)C1)=O)(CC(F)(F)F)NC(c1c(CC)noc1C)=O C1(NC(C=CCOC)=O)CCCC2CN(C(=O)COc3ccccc3SC)CC12 N1(C(C(CNC(C(CCC)NC(N)=O)=O)(C)C)=O)CC2C(C1)C2(C)C C1(C(=O)NC(C)CN2CCCC2)C2CC2CN1C(c1csc(O)n1)=O c1(C(CCC)C)nc(-c2cc(SCCO)nn2CCC)n(C2CCSC2)n1 Cc1ccc(CN2CCCC(C(N3C4CCC3COC4)=O)CC2)c([N+](=O)[O-])c1 CC1CCn2cc(C(=O)NC(CNC(=O)C(F)(F)CNC)CO)nc2C1.N(C)C Cc1nn(C(C)C)c(C)c1C(N1CCOCC(NC(=O)CC2CN(C)C2)C1)=O C1(NC(CC2CCN(C)C2)=O)CC2CC(NC(c3nc(Cl)cs3)=O)CC12 c1(C(N2CCC(CNC(CCc3c(C)nn(C)c3)=O)C2)=O)cc(Br)c(C)cn1 N12CC3(CO)CC1(C3)C2=O.C1(C)(NC2(CC(=O)OC)CC2)CCCC1O.C(C)=O C1(C(N2C(COC)(CNC(=O)Cc3csnn3)CCC2)=O)CCC(=O)CC1(C)C C1(C2CCCCN2C(=O)C2CC2)(CNC(=O)CCc2nccs2)CCOCC1 c1(C(C)=O)cc(C(N2CCC(CO)(NC(C34CCC3C4)=O)CC2)=O)c(C)nc1C C1(C(=O)NC(CCCC)C)N(C(=O)CSCCC(C)C)CCC1(C)C C12(NC(c3cccc(SC(F)(F)F)c3)=O)CC(C1)N(C(c1cncc(O)c1)=O)C2 c1(C(=O)OCC)cc(N2CC(CNC(C3CC34CCCOC4)=O)C2)oc1[N+](=O)[O-] C(CN=c1nc2ncn(C)c2c(NCC2CCS(=O)(=O)C2)[nH]1)(C1CC1)NC(=O)NC c1(C(=O)NC2C(NC(C(C)N(C3CCC3)C)=O)CC2)cccc(-n2ccnn2)c1 c12cccnc1C(=O)N1C(CC1)C(=O)N2.c1(C)ccnn1CCO.c1(N)cscn1 Cc1ccnc(O)c1C(=O)NC(CNC(=O)C(C(C)C)n1cnnc1)C1CC1 C1(CCC(=O)N(CCN(C(=O)C(CO)NC(N)=O)C(C)C)C)CC(F)(F)C1 C1(NC(C(C)OCC)=O)CN(C(c2cc(C)c(CC)nc2O)=O)CC1N=[N+]=[N-] c1(CC(=O)NC(C)CNC(=O)Cc2cnco2)ccc(C2CCC2)cc1 C#CC(C)(C)C(=O)NC(CC)C(=O)NC1CCCCC1C(=O)NC1C2CN(C)CC12 N1(C(CC(=O)OCC)=O)CCOCC2(C1)CN(C(C1CCCC1)=O)CCCO2 C(CC(CC)C(=O)NCC1(CNC(c2cnc(Cl)s2)=O)CC12CCC2)=CCCC C1(NC(C2CC(C)(O)C2)=O)CC2CCC1CN2C(C1CCCN(C(=O)N(C)C)C1)=O C12(C(=O)NCC(CCNC(c3cnc(CCC)s3)=O)OC)CCCC1C2(F)F C(N=c1nc2[nH][nH]cc-2c(O)n1)C1(C)CCN(C(c2c(CC)onc2C)=O)C1 Cc1ccc(C(N2C3CCC2CN(C(C2CCN(C)C2=O)=O)C3)=O)c(N)c1Cl C(=O)(C1CN(C(=O)NC(CCC=C)C(=O)OC(C)(C)C)Cc2n[nH]cc21)OC c1(CC(=O)NCC(COC)N)cc2c(cc1Br)OCCO2 CN1CC2CCN(C(=O)CCN(CCCO)C(=O)CC3CCCOC3)CC2C1 CC(c1cnn(C)c1)=CC(N1CCN(C(C2CSCC(=O)N2)=O)C(C(F)F)C1)=O c1(CCC(=O)NC(CNC(Cc2cnc(C)s2)=O)CC(C)C)ccc(Cl)c(F)c1 c1(C(=O)NCCCN(C(C2CC(C)=C(C)CC2)=O)C)ccc2n[nH]cc2n1 c1(NC(C)=O)cccc(F)c1C(N1CC(O)(CN(C)C(C2CCS2(=O)=O)=O)C1)=O C1(NC(c2ccc[nH]2)=O)CC2CC(NC(C3CCCC4(CC4)C3)=O)C1C2 N1(C(CCNC(c2cc(C(C)C)no2)=O)=O)CCC2CCCCC12 N1(C(C2CN(Cc3ccc(COC)o3)CC(F)C2)=O)CCN2CCOCC2C1 N1(C(c2c(C)ncnc2)=O)CCC(CNC(c2cncn2C)=O)C(C)C1 c1(OC)ccc(C(=O)NC2CCCC2NC(c2c(C)nn(C)c2Cl)=O)c(F)c1 c1(OC)ccnc(F)c1C(N1CCC(O)(C(C)NC(=O)CCC(F)(F)F)C1)=O c1(NC(c2ccnc(F)c2Cl)=O)cc(Cl)c2cn[nH]c2c1 C1(C)(CNC(C(C)(C)C2CCC2)=O)CN(C(C2(C)CCCO2)=O)CCO1 Cc1ccc(Cl)c(NC(=O)C(N2CCC(C(C3CC4CCC3C4)N)CC2)=O)c1 N1(C(CCC(=O)N(C)C)=O)C(CC(=O)NCc2ccnc(Cl)c2)C2CCCC12 C12(C(=O)NC(C3CCN(C(c4ccn(C(C)(C)C)c4)=O)C3)C)CC=CC(C1)OC2 CCC(C)(C#N)C(=O)Nc1ccc(NC(=O)C(O)C(F)(F)F)c(C)c1 CN1CCCN(C(C23CC(CO2)N(C(=O)CN2CCSCC2)C3)=O)CC1 N1(C(C(Cc2ccco2)NC(c2c(C)cns2)=O)=O)CC2(CNC(=O)N2)C1 N1(C(C(C)CCN2CCOCC2)=O)CC(c2ccccc2)CCC1C Cc1onc(C(=O)NCC2CCN2C(=O)CCC2CC2(C)C)c1[N+](=O)[O-] c1(C(=O)OC(C)(C)C)cc(C(=O)NCc2ccc(-c3nnco3)cc2)cc(Br)c1 CC1(CNC(=O)C(F)=C2CCC2)CCCN(C(=O)C(c2cccc(F)c2)O)C1 C1(CNC(c2cc(OC)n[nH]2)=O)CCCC2CN(C(=O)Cc3cc[nH]n3)CC12 C1(O)(CC(=O)N(CCNC(=O)C(F)C2CCCC2)CC)CCC1 c1(C(N2CCCC(CC(=O)Nc3ccc(C4CC4)nc3)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CS(=O)(=O)CCC(=O)N1CC2CC(NC(=O)C=CCN(C)C)CC(C2)C1 c1(C(=O)NCC(C)N(C(C(C)NC(CC)(C)C)=O)C)cc2ccccc2c(O)n1 c1(C(=O)NCC(CN(C(=O)C(C#N)C2CC2)C)(C)C)cccc2c1OCCC2 C1(N(C(C(C=C)C)=O)CC=CCCCCC)CCN(C(=O)COC(C)CC)CC1 N1(C(C2(C#C)CCC2)=O)CCCC(CN(C)C(C2(OC)CS(=O)(=O)C2)=O)C1 c1(N(C2(CC)CCC2)C)nnc(CCCC2CCOCC2)n1CCC#N.N CCC(C(=O)NC1CN(C(=O)C(F)F)CC1(C)C)C(C)O c1(N2CCC(NC(C(=O)N(CC(O)CO)CCC)=O)C2)ncccc1O C1(C(N2CCOC(c3ccc(C(F)(F)F)cc3)C2)=O)CCC12CCC2 C1(C(=O)Nc2ccccc2)(CC2(OC(c3onc(C)n3)C)CC2)CCCC1C C1(NC(C2CC3CC3C2)=O)CCCN(C(C2CC(=C3CC3)C2)=O)C1 N1(C(c2nnc(C(C)(C)C)s2)=O)CCCCC(NC(c2csc3cncn23)=O)C1 c1(C(=O)NCC2(CC(=O)NCC(C(=O)NC)C)CC2)cc(C)c(C)o1 N1(C(C2CC3(C(OC)CC3)C2)=O)CC2CCN(C(c3ccc[nH]3)=O)CC2C1 N1(C(Cc2c(C)ocn2)=O)CCCC(F)(CNC(=O)CN2CCSCC2)C1 C1(NC(Cc2c(C)scc2)=O)CN(C(C2CCN(C)C2)=O)C2(CCC2)C1 N1(C(C2C3CN(C(C(CC)COC)=O)C2C3)=O)CC2CN(C)CC2C1 C1(NC(C2C(OC)CC2)=O)CCN(C(=O)CCN2CCCCC2=O)C12CC2 C1(C(N2CCC(CCN(C(CSC)=O)C)CC2)=O)CCc2nc(C)cn2C1 c1(C(C)=O)ncc(C(=O)NCCC(C)N(C(=O)C=C2CC2)C)s1 N1(C(CC(C)C)=O)CCC2CN(C(=O)CCCc3ccc([N+](=O)[O-])cc3)CC2C1 C#CCCCCC(=O)NC1CCN(C(c2ccc(N)c(O)c2)=O)C1 C=CC1CCN(C(c2nc(CNC(c3cc(CC)no3)=O)oc2C)=O)C1 C(=O)(CC(F)(F)C(C)C)NCCN(CCC)C(C1CCOCC12CCC2)=O C(CCCC(=O)NC(C(=O)Nc1cnn(C)c1C)C1CCOC1)SC c1(C(=O)OC(CC)C(N)=O)cc2c(s1)CCN(C(=O)OC(C)(C)C)C2 c1(CC(=O)NCC2C(NC(Cc3nc(C)sc3)=O)C2)cccc(C(F)(F)F)c1 n1(CC(N2C(CC(=O)NCc3ncc[nH]3)COCC2)=O)ccc2c(F)cccc12 C1(CNC(C(F)=CC)=O)CC(C)(C)CCC1NC(=O)CS(=O)(=O)CCO C1(C(=O)NC(C)(C)CC2CCCC2)C(C2CC2)CCN1C(C1CS(=O)(=O)C1)=O C(=O)(CCC(O)C(C)(C)C)N1C(CN(C)C(c2cn3c(n2)CCC3)=O)CCCC1 C1(c2cn(C3C=CCCC3)nn2)(NCC(=O)N(C)Cc2cncnc2)CCCOC1 c1(C(N2C(C(=O)NCC(=O)NC(CC)CO)CCC2)=O)ccc(C#N)cc1SC c1(N2CC(CC(C)NC(C3CCCN(C(C)=O)C3)=O)C2)ncc(C)c(C)n1 C12(C(=O)OC)CC1CN(C(=O)CC1CN(C(=O)CSc3cn[nH]c3)CCO1)C2 CCCC(CC)C(=O)NC12COC(C1)C(NC(=O)COCc1nccn1C)C2 c1(C(=O)NC2C=CC(CNC(Cc3nc(CC)sc3)=O)C2)ccc(C#N)[nH]1 C(C(=O)NC1CCC(CCCN2C(C)CC2(C)C)C1)(C(C)C)SCC c1(NC(C(CC#C)(C)NC(=O)C(C)OCC2CC2)=O)cc(C)cn(C)c1=O N1(C(C2(C)CCC(=O)NC2)=O)CCN(C(c2ccc(N)c(Cl)c2O)=O)C2CCC12 CN1CCN(C(C2CCN2C(C2CC23CC3)=O)=O)Cc2ccccc21 N1(C(=O)C=C2CCCCC2)CCN(C(C2C3CCC(=O)C23)=O)C2CCCC12 c1(C(N(CC(C)(C)NC(C2N(CC)C(=O)CC2)=O)C)=O)cc(=O)c(Br)c[nH]1 C1(C)(CC)CC(NC(=O)CC(=O)N(C)C)CN1C(c1ncnn1CC)=O N1(C(C(c2ccccn2)C)=O)CCC(C)(CNC(C2CN(CC(F)(F)F)C2)=O)C1 C(CS(=O)c1ccc(CC(=O)NCCN(C(=O)C2=C(C)OCCS2)C)cc1)OC C=C(C)CCC(=O)NCC1(CNC(=O)Cc2csc(CCCCC)n2)CCC1 C1(N(C)C(c2csnc2Br)=O)C2CN(C(=O)CCC3CC3(C)C)CC12 N1(C(c2nc(C)sc2C)=O)CCC2CCCC(C1)N2C(c1c(C)cncc1C)=O c1(-n2ncc(C(=O)NC(CNC(Cc3c(C)n[nH]c3)=O)C)c2)ncc(Cl)cn1 C(=O)(CC(C)(O)CC(=O)O)N1C(C(=O)Nc2c(F)ccc(C)c2Cl)COCC1 N1(C(C2CC(NC(c3c[nH]c(=NC)s3)=O)C23CCC3)=O)CCCCC2(CCC2)C1 C1(NC(C(C)N(C(C(N2CCOC2=O)C)=O)CCO)=O)CC2CC1CC2CO c1(C(=O)NC2CCCC(CNC(COCC#C)=O)C2)c(C)nn(C)c1Cl C1(C(=O)NC(C)CSCCO)(COC)CN(C(=O)Cc2ccccc2)C1 C1(N(C(c2cc(CCNC(CCOCC(C)C)=O)on2)=O)C)CCC(=O)N(C)C1 CC(O)C(C(=O)NCC1(F)CC(NC(c2cc[nH]c2)=O)C1)NC(=O)C(F)(F)F Cc1[nH]nc2ccc(C(N3CC4(CCN(C(C5CCCOCC5)=O)C4)C3)=O)cc12 C(=O)(CC(C)C(F)F)NCCC1(NC(c2occ(C)c2)=O)CCCC1 c1(C(C(=O)NC(C)C(C)NC(C2(n3cncn3)CC2)=O)C)ccc(F)cn1 C(=O)(C1COc2ccc(Cl)cc21)N1CCCC(CNC(C2(C)CC2)=O)(CO)C1 c1(C(=O)NC2C(CNC(C3(OC)CC3)=O)C2)ccn(CCO)c(=O)c1 C1(C(=O)NC2C(N(C)C)CCC2)CCCN(C(C2(F)CCOC2)=O)CC1 c1(C(=O)NC2CCSC23CN(C(C2(CCO)CC2)=O)C3)ccc2c(c1)CCOC2 C1(CC=C)(NC(=O)Cc2ncoc2C)CCN(C(C2(n3cccn3)CCC2)=O)C1 C(=O)(C(F)C(C)CNC(=O)Cc1ccon1)NCCn1c(C)cnn1 C(C(N=[N+]=[N-])C(=O)N1CC(C(=O)NC(CO)CCF)(SC)C1)OCC C1(C(N(C2CSC2)CC#C)=O)CCCN1NC(=O)C=CC(C)(C)C N1(C(c2ccc(CC)o2)=O)CC(N=c2[nH]nc(C(F)F)s2)C2(CCC2)C1 c1(C(=O)NC2C(NC(C(c3cccc(OC)c3)O)=O)C2)cccc2ncsc12 Cc1ccc(SCCC(N2CCC(CO)(NC(C3C4CCC3CC4)=O)C2)=O)cc1 N1(C(CCN(CC)CC)=O)CC(CNC(c2ccc(CO)cc2)=O)C2CC12.C(C)(C)O CCCC(CNC(c1c[nH]nc1C(F)F)=O)C(=O)NC(c1ccncc1)C Cc1nc(C(C)C)ccc1NC(N1CCOC(C(C)O)C1)=O N1(C(C(C)(CO)OC)=O)CC2CCC(C1)N2C(=O)C[SH](c1ccc(O)cc1)C.C1CC1 N1(C(c2ncc(OC)cn2)=O)CCCCC(NC(=O)C=C(F)c2ccccc2)C1 C1(NC(C2C(OCC)CC2)=O)CCCC1(C)CN(C(=O)CC1CCCCN1C)C C(=O)(C(C(C1CC1)C1CC1)N(c1c(C)nc(C(=O)OC)o1)C)OC c1(NC)ccccc1C(=O)NCC1CC(O)(CNC(c2cc(C(N)=O)no2)=O)C1 C1(C(=O)NCCC(C)N(C(c2ccc(SC)o2)=O)C)CC2OC(=O)OC2C1 N1(C(c2c(C(C)O)cccc2)=O)CC2CCC2(CNC(C2(C(F)F)CC2)=O)C1 c1(OC)cc(F)ccc1CC(N1CC(N(C)CCl)C(C(C)C)C1)=O N1(C(c2oc(CC)c(C)c2)=O)CCCC(C)(C)C1C(=O)NC(C)C(C)F c1(C(=O)NCCN(c2ncc(C(F)(F)F)cn2)CCOC)c(C)cnn1C c1(OC)cc(CNS(=O)(=O)CC(C)C#N)c2c(c1)CC(C)O2 Cc1ccc2ncnc(N3CCC(NC(c4nccn4C)=O)C(O)C3)c2c1 c1(C(N(CCCOCCNC(C(C(CC)C)C)=O)C)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)N(C2(CNC(c3[nH]n(C)c(=O)n3)=O)CCCCC2)C2CC2)cc2c(s1)CCC2 CCC(CC(F)F)C(=O)NC1CCC(CNC(C23CC(F)(C2)C3)=O)CC1 Cc1cc2cccc(C(N3CCN(S(=O)(=O)c4ccccn4)C4CC34)=O)c2[nH]1 c1(C(=O)NCCN(C(CCC(C)SC)=O)CC(C)O)cnc(C)c(N)c1 CC(C)C(C(=O)NC(C)C(CO)NC(C1(O)CC(F)(F)C1)=O)n1cnnc1 C1(CNC(C(C)O)=O)(NC(=O)CS(=O)(=O)N2CCCCC2)CCCCC1 CC12CC(C(=O)NC3CC(O)CN(C(c4ccc(CO)s4)=O)C3)(C1)C1(COC1)O2 C(=O)(CC(C)C(C)(C)C)N1CC(C(=O)NCCn2c(C)cnn2)C(C)(C)C1 c1(NC)c(C(N2CCC(N(C(=O)C(C)=CC(C)(C)C)C)C(C)C2)=O)cccc1F c1(C(c2nnnn2Cc2ccccc2)NC(c2ccccc2)CC)coc(C)n1 Cc1oc2cc(C(N3CC(C)(NC(C4CCCCS4)=O)C3)=O)[nH]c2c1C Cc1nnc(C(=O)NC2CC(F)(CNC(c3cccn3-c3ccccc3)=O)C2)s1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(CCNC(C=CC(=O)N(C)C)=O)CC1 Cc1cc(Cl)c(F)cc1C(=O)NC1CC1C(=O)Nc1ccc(C#N)cc1C(F)(F)F C1(CC(=O)N(CC(N2CCN(C(=O)NCC)CC2)=O)C)CCC2(CC1)CC2 c1(C(=O)NC(CCCNC(C(CCC)NC(N)=O)=O)C)ccc([N+](=O)[O-])c(SC)c1 C1(C(C)(C)C)COCCN(c2nnnn2C(c2ccc(Br)s2)C)C1 c1(CN(C)C)cn2cccnc2n1.C123CCCN(C1C2)C3=O C1(NC(c2cn(C(C)(C)C)nc2)=O)CC(CNC(c2ccns2)=O)CC1O CN1CCC2CN(N3C(C4(C=O)CC4)CCC3)CCC12.C1(CC(=O)NC)CC=CC1 c1(C(N2C(CCNC(COC)=O)C(C)CCC2)=O)cc2c(C)cc(F)cc2[nH]1 c1(-n2cc(CSC(C(CO)NC(C(=O)NC(C)C)=O)C)nn2)cccc(F)c1Br C(=O)(C1=C(CCCCl)N(CC2CC2)C(=S)NC1c1ccc(OC)s1)OC C(=O)(CC(C)(CN)C(F)(F)F)Nc1cncc(-c2cccc(C)c2)c1 N1(C(CC=CCCCCC)=O)CCC(C(=O)NCCCO)(CCOC)C1 C1CC(O)C(=O)N1.Cn1cncc1C1CC1C(N1CCC(N2CC(O)C2)C1)=O C1(C(=O)OC)CN(C(=O)C(=O)NCc2nc(=O)n(C)[nH]2)c2ccnn2C1 n1(C(CC)CC)nc(C(=O)NCC=CCNC(c2onc(Br)c2C)=O)cc1C O=C(N=c1cco[nH]1)c1scnc1CN1CCN(c2ccc(F)cc2)CC1 Cc1nc(C(N2CC(N(C)C(c3cc(Cl)cn3C)=O)C(O)C2)=O)ccc1[N+](=O)[O-] c1(C(N(C2CCCN(C(CCCNC(C)=O)=O)C2)C)=O)cnc2ccnn2c1 C1(NC(c2n(C=C)nnc2)=O)CCC12CN(C(c1ccc(OC(C)C)nc1)=O)C2 C#Cc1cnc(C(=O)N(CC(=O)NC2C(C)C2(C)C)C)c(C)c1 c1(OC)ccc(CCCCC(=O)N2CCC(CC(C)NC(=O)C(C)O)CC2)cc1 c1(C(N(CC(C)NC(CCCC(C)O)=O)C)=O)cc(Cl)cc2c1NCCC2 S(=O)(=O)(c1cc(C=CC(=O)NCC(c2ccccc2)C)ccc1OC)COCC c1(C(N2CC(CNC(=O)C(F)OC(F)(F)F)C(O)C2)=O)cc2c(s1)CCC2 C1(C(=O)NCC2CC(F)(CNC(CNC(CC)=O)=O)C2)(C(F)F)CCOCC1 c1(CC(N2CC(=C(CNC(C3CCCCO3)=O)F)C2)=O)ccc(F)c(Br)c1 C(=O)(CCC(F)F)N(C(CNC(C1CCCC1(C)C)=O)C1CC1)C C(CNC(c1cc(C2CC2)n[nH]1)=O)(CC(=O)N(C)CCN(C)C)OC c1(C(=O)NC2C(NC(C3CC(C)OC(C)C3)=O)COC2)c(Cl)ccc(F)c1F Cc1cc(F)ccc1C(=O)NCCCCc1cn(-c2ccc(F)c(Br)c2)nn1 C1(C2CCCCO2)(C(=O)OCc2cn(CCCC)nc2C)CCCO1 c1(C(=O)NCC(c2cc(F)cc(Cl)c2)NC(C(C(C)C)C)=O)cccc2ncnn12 C(=O)(C(C)c1cc[nH]n1)N(CC(=O)NCCOCCCC)C1CC1 n1(CC)cc(C(N2CCC(C(F)C(N3CC(C)(O)C3)=O)C2)=O)nn1 c1(CC2(C(=O)NC(CNC(c3nc(C)oc3)=O)C)CC2)cccc(F)c1F N1(c2cccc(OCCCOC)c2)CC2CN(c3ncncc3F)CC2C1 c1(C(=O)OC)ccc(C(=O)OCC2CCCO2)c(Cl)c1.C12CC(C1)NC2=O C(C(N=[N+]=[N-])C(=O)N1CCN(C(=O)COC2(C)CCC2)C(C)C1)OCC CC(C)C(O)C(C)C(=O)N1CCN(C(=O)C(C2(O)CCCC2)F)CC1 C1(C(N(C(C)CNC(=O)Cn2c(C)ccc2C)CC)=O)COC(C)(C)CO1 Cc1sc(-c2ccco2)nc1C(=O)NC(C)CNC(c1cc(CC2CC2)on1)=O C1(NC(=O)C=CBr)CCCN(CCCNC(=O)CNC(c2ccc(F)cc2)=O)C1 N1(C(c2cc(C)oc2)=O)CC2CC1CC2NC(c1cc(C)oc1C(F)(F)F)=O C1(CC)CN(C(=O)C(=O)NCc2ccc(Cl)cc2)CCC1=O c1(C(=O)NC(CCCNC(c2n[nH]c(CC)c2Cl)=O)C)cccc(Cl)c1N C1(C(=O)NCC2CCN(C(=O)Cn3cc(CO)nn3)C2)Cc2cscc2C1 N1(C(CCNC(C(COC(C)C)OC)=O)C)CCNC(=O)C1 N1(C(C(=O)NN2CCOCC2)CC2CC(OC)(OC)C2)CCC(F)(CF)CC1 N1(C(C)C)CCCCC1NC(COC(C1CC(C(=O)NC(C)(C)C)C1)=O)=O.C1CCC1 C12CC(C13CCC3)CO2.Cn1ccc(NC(=O)COCCCF)n1 C(N1CCC(S(=O)(=O)NCc2ccccc2)C1)n1nnn(C2CCC(C)O2)c1=S C(=O)(CN=c1cc[nH]cc1)N1CC(CNC(c2c(CN(C)C)cco2)=O)C(O)C1 c1(OC)cc(Cl)c(Br)cc1C(=O)NCC(CO)NC(C1(Br)CC1)=O Cc1noc(C2CC2)c1C(=O)NC1CCC1NC(=O)CC(O)CN(C)C CC1CC(=O)CC(C2CCCCC2)N1C(=O)CSc1cn(CCCF)nn1 C1(C)(CC)C=C(C(=O)N2CC3CC2CN3C(c2ncsc2Br)=O)C1 N1(C(C2(C=C)CCC2)=O)CC(CNC(c2csnc2C2CC2)=O)C2(CC2)C1 c1(OC)cc(C(N2CC(NC(=O)C(C)(C)c3cncs3)C(O)C2)=O)cc(Cl)c1O C#CCCCCCC(=O)N(CC(C)(C)C(=O)NC1CCCC1C#C)C C(C1(O)CCCc2ccccc21)NC(=O)NCCC12COC(CO1)C2 c1(CNC(C2CN(C(C)=O)C2)=O)nccc(C)c1F.C12(CC(F)(F)C1)C(=O)N2 CC1(C(=O)NCCOCC(=O)NC2CCCSC2)CCC(=O)C1 Cn1nc(C(N2CCCC(Cn3cc(CSC4(C)CC4)nn3)C2)=O)cc1C1CC1 N1(C(CS(N)(=O)=O)=O)CC(NC(c2cc(O)cnc2Cl)=O)CC12CCC2 N(C(=NCc1ccnc(C(F)(F)F)c1)NC1CCC1)C(C#C)C C1(C(=O)NCC2N(C(C(CC)C)=O)CCCC2(C)C)CC(c2cnn(C)c2)=NO1 c1(C(=O)NC2(COC)CCOCC2)cc2ccc(Cl)c(S(=O)(=O)NC(C)C)c2s1 Cc1nc(Cl)nc(N2CCCC2C2CCN(C(C3CC=CC3)=O)C2)c1Cl C(=O)(CCCCCN=[N+]=[N-])NC(C1(O)CN(C(c2cc3ncccc3[nH]2)=O)C1)C c1(CNC(=O)CCc2ccncc2)cc(O)nc(CNC(C2(C(N)=O)CC2)=O)n1 C(=O)(C1=Cc2cccc(OC)c2OC1)NCC12N(C(CC)=O)CCC1CC2 C1(NC(CN(CCC)C)=O)CC2CCC1C(NC(c1cc3c(ccn3C)[nH]1)=O)C2 Cc1ncnc(N2CCC(NC(C3(c4ccc(Cl)cc4)CCC3)=O)C(O)C2)c1Br C(=O)(C1CSc2ccccc21)NC(CNC(c1csc(C)c1C)=O)CO Cn1c(=N)[nH]c2cc(C(=O)NC3COC4(CCCN(C(=O)CNC=O)C4)C3)ccc12 c1(C(N(C)CC2(NC(C3C(CC)OCC3)=O)CC2)=O)ccnc2ccc(O)cc12 N1(C(c2nn(C)c(Cl)c2)=O)CCC2(CCCN(Cc3cccc(I)c3F)C2)C1 C1(NC(N2CCCC(C)(C(=O)O)C2)=O)CNCC2(CCC2)C1 C1(NC(C(CC)CCOC)=O)CCCCCN(C(=O)Cc2cc(C)cc(C)c2)C1 c1(C(=O)NC2CC(C)N(C(=O)Cn3cnnc3)C2)ccc2ccc(Br)cc2n1 N1(C(c2cccc(C)c2O)=O)CC(NC(C2CN3CCN2CC3)=O)C2(CCC2)C1 C1(CNC(c2ccc(C)cc2)=O)CCC(C)CN1C(=O)CCOC(C)C C(=O)(C(C)(O)C(C)(C)C)N1CC(COC)N(C(c2ccc(F)c(SC)c2)=O)CC1 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)Cc2c(F)cccc2Cl)CC1CC1CC1 CCCC(C)CC(=O)N1CCC(F)(CNC(c2ccc(COC)[nH]2)=O)C1 c1(C(=O)NCC(C)N(C)Cc2cnsn2)cc(-c2ccsc2)nn1C N1(Cc2nc(C(=O)NC)n(C)n2)CCC(=O)N(CCN(CC(C)C)S(C)(=O)=O)C1=O N1(C(C2CC(C)(C)OC2)=O)C2CCC1CC(NC(c1cc(Cl)cc(F)c1F)=O)C2 Cc1noc(C)c1S(=O)(=O)N1CCC(O)(c2nc(-c3ccc(Cl)cc3)no2)C1 C(CCC(O)C(=O)NCCn1cnnc1)NC(CCC(=C)Cl)=O CC1CCC(C)(C)CN1C(=O)C(=O)NC(c1ccc(F)cc1)c1cn(C)cn1 c1(C(N(CCNC(CC2CC(=C)C2)=O)C(C)C)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 N1(C(C(=O)NCCC)=O)CCN(N2CC(C(=O)OC(C)(C)C)C3(CCC3)C2)CC1 N1(C(c2ncn(C)n2)=O)CCCCCC(NC(C2CC(n3cnnc3)C2)=O)C1 C1(C)(CNC(C(CC)(C)NC(C)=O)=O)CN(C(=O)CCOC(=O)NC)CCO1 C1(CN(C(C2C=CCCC2)=O)CC)CCCN1C(=O)C(C)N1CC(OC)C1 N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2(CCCN2C(C2CCSCC2)=O)C1 c1(C(N2CCC(CC=C)(NC(=O)Cc3cnc[nH]3)C2)=O)cnc(Br)c(OC)c1 c1(C(N2CCC(NC(C3(SC)CCC3)=O)C2)=O)cccc(Br)c1 N=c1ncc(C(=O)NC2CCCCC2NC(c2cocc2Br)=O)c[nH]1 C(=O)(C(CNC(CC(C)C)=O)CO)N(C(CCNC(=O)OC(C)(C)C)C)C.C(N)(=O)N c1(C(C)=O)ccc(C(N2CCCC2(C)CNC(=O)COC2CCCCC2)=O)nc1 C(=O)(CC(C)(C)C(C)=O)NC(C(=O)N(CC(CC)N)C)C(C)OC.OC N1(C(C(CCC(C)C)NC(C2CN(CC)C(=O)C2)=O)=O)CCCC2CCCCC12 c1(CN(C(C)=O)CCNc2cccc(Br)c2C)cc2c3c(c1)CCCN3CCC2 C1(NC(C2CC(n3cccn3)C2)=O)CCN(C(c2cnco2)=O)CC12CCC2 c1(NC(C(N2CC3CCC2C(O)C3)c2nc(C)c(Br)s2)=O)ccc2c(c1)CCC2 C1(C)(NC(C)=O)CCN(C(=O)C(c2ccoc2)NC(=O)CC2CCCCC2)C1 C1(C(N(C)CC2N(C(COCCOC)=O)CCCC2)=O)NC(=O)C2CCC12 C1(CNC(c2c(C)cncn2)=O)CC2(CCC2)CN1C(=O)CSCC#N Cc1nccc(C(=O)NCCCC(C)(C)NC(C23CCCCC2C3)=O)c1N C1(NC(Cc2cnc(C)s2)=O)CC=C(C(=O)NCC(C)(O)CO)C1 N1(C(CC=C)=O)CC2CCN(C(c3cc(-c4ccn(C)n4)on3)=O)C(C2)C1 C1(CC(=O)Nc2ncn(CC)n2)CCCN(C(=O)C(C(C)C)OCOC)CC1 C(CCC=CC)(C(=O)NC1CCC(F)(F)CC1)N(CCSC)CC N1(C(CS(CC)(=O)=O)=O)CCN(C(=O)Cc2ccc(C)cc2Cl)C(C)CC1C CC1(C)C2CC(NC3CNC4(CCC4)C3)CC12 c1(C(N(C(C)CNC(=O)C(C)(C)n2cnnn2)C)=O)cnc(N)cn1 C(=O)(CCCCC(=O)N(C)CC1(O)CN(C(c2ccnn(C)c2=O)=O)C1)OC C(=O)(C1=NOC2COCC12)N1CC(NC(Cc2cccc(CC)c2)=O)C1 c1(NC(C2C(C)CN(C(=O)C(C3CC3)N(C)C)CC2)=O)cccc(N=[N+]=[N-])c1 C1(CC=C)(NC(=O)CC2CC=CC2)CCCN(C(C2CCN2C(C)(C)C)=O)C1 CC(C)(C)CC(O)C(=O)NC1CN(C(c2sccc2-n2cnnn2)=O)CC1O C1(NC(=O)C(F)=CCCF)CC(O)CN(C(=O)C(C2CCCCCCC2)O)C1 c1(OC)cncc(C(=O)NC(C)C(C)NC(=O)CCCn2cncn2)n1 N#CC1CCCC1NC(=O)CC(CC1CC1)NC(c1ccncc1)=O Cc1noc(N)c1C(=O)NC(CCN(C)C(c1cncn1C1CC1)=O)C(C)C c1(OC)cnc(C(=O)NCC2C(C)CCN2C(=O)CCc2ccsc2)cn1 Cc1ccc2cc(C(N3CC4CC3CN4C(=O)CC3OCCCO3)=O)ccc2n1 C1(N(CC(F)F)C(C2(CC(C)=O)CC2)=O)CCOCC1 c1(C(=O)NC2C(F)(F)CCN(C(C3CN(C)C3)=O)C2)nc2ccc(F)cn2n1 c1(C(N2CCCC(N(c3ccc(C)cn3)C)C2)=O)cncc(P(C)(C)=O)c1 C(C)(C)(C(C)CC(=O)NCc1cnn(C)c1O)NC(C(CC#C)C1CC1)=O N1(C(CCC=CC)=O)CCCCC1C(C)NC(c1cn(-c2cccnc2)nn1)=O C(=O)(C1=CC2CCC(C1)C2)N1CCCC(CN(C(=O)CC2CC2)CC)C1 Cc1ncn(C)c(=O)c1C(N1CC2CC2(NC(=O)CC2CC3(CC3)CO2)C1)=O n1(CC(N2CC(CC)C(NC(=O)C(C(C)C)N(C)C)C2)=O)cccc(C)c1=O CC(C)CC(CNC(C1(c2cc[nH]n2)CCC1)=O)NC(=O)Cc1cscn1 c1(NC(C2CC(F)CN(Cc3ccnc(O)c3)C2)=O)cc([N+](=O)[O-])cc(Cl)c1O N1(C(c2ccc(OC)o2)=O)CC2CN(C(C3CS(=O)(=O)C3)=O)CC(F)(F)C2C1 C(=O)(CCC(C)(C)NC(=O)C(C)CN(C)C)NC1(COC)CCOC1 C1(C(C)C)CN(C(=O)CCC(C)C#N)CCCN1C(=O)C=Cc1cccc(Cl)c1 n1(CC(N2CCC3C(NC(CC4N(CC)CCC4)=O)C32)=O)cccc(N)c1=O N=c1[nH]c(N2CCn3c(cnc3Br)C2)nc2ccc(Br)cc12 C(=O)(CN=c1ccc(C#N)c[nH]1)NCC1C(CNC(c2c(C)cc(C)nc2)=O)C1 C1(C(=O)NCCN(C)C(c2cnsc2)=O)C(c2ccccc2)C1(C)C Cc1cc(=NCC2CCCC(F)C2)[nH]cc1S(=O)(=O)N(C)C(C1CCCCC1)C Cc1cc(F)ncc1C(=O)NC(C)CC(C)NC(C1(CF)CCC1)=O Cc1cc(Br)cc2cc(C(=O)N(CC(C)CNC(=O)CC(C)(C)C#N)C)[nH]c12 CC1Oc2ccc(C(N3CCC4(CCC4)C3)C(=O)NC3CCCC3)cc2NC1=O c1(C(C(=O)NC2(CCNC(C(CC)NC(N)=O)=O)CC2)C)ccc(F)c(F)c1 N1(C(C2C(CC)CCO2)=O)CCC(O)(CNC(c2cc(C(F)F)no2)=O)C1 c1(CC(N2CCCCC2CN2CCCC2)=O)cccc2ccncc12 N1(C(c2c(C)ncnc2)=O)CCC2(CC1)CN(C(c1ncc(N)nc1C)=O)C2 c1(CCCC(N2CCC(O)(CNC(CCCC#N)=O)C2)=O)c(F)cccc1F N1(C(CCn2c(C)nc(C)n2)=O)CC(F)(F)CC1CNC(C1(Cl)CC1(F)F)=O c1(CCC(=O)NC(C2CCCN(C(COC)=O)C2)C)cc(OC)ccc1OC C1(CNC(C2(SC)CN(C(C3CC(=C4CCC4)C3)=O)C2)=O)CCCCN1C C1(C(=O)N(CC(F)(F)F)CCO)CN(CC2CCC(O)CC2)CCO1 c1(C(=O)NCC2C(OCC)CN(C(=O)C(C)(C)OC)C2)cc2c(C)noc2s1 C(=O)(C(CC(=O)OC(C)(C)C)SC)NCCOC.C(CC(=O)NCCSCC)NC S(=O)(=O)(c1c[nH]ccc1=NC(CO)C1CC1)NC(CCOC)Cc1ccco1 c1(C(N(C(=O)C(c2ccccc2)OC)CCC)C)ccccc1O c1(NC(=O)NC2(SCCCN3CCS(=O)CC3)CC2)cccc(Cl)c1Cl C1(C)(CN(c2cc(CNC(=O)OC(C)(C)C)c(Cl)cn2)C2CC2)CC(C2CC2)=NO1 CN1CC(C)(C(=O)NCCCC2CN(C(C3(CO)CC3)=O)CCO2)CC1=O C1(N(C(=O)CCc2ccsc2)CC)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 Cc1cccc(N(C(=O)CNC(CCc2ccc(-c3nnc(S)o3)cc2)C)C)c1 c1(C(=O)NCC=CCNC(c2ccc(C)c(C)c2)=O)ccc(N)c(C)c1C N1(C(CCc2scc(C)c2)=O)CCC(C2(NC(=O)CCn3cc(Cl)cn3)CC2)C1 C1(CNC(C(CSC)(C)C)=O)(NC(c2ccc(C(F)F)o2)=O)CC2CCC1CC2 c1(C(N2CCC(C)C(N(C)C(c3cn[nH]c3)=O)C2)=O)nccc2n[nH]cc12 C1(C(=O)NCC2CCN(C(c3nc(C)c(C)[nH]3)=O)CC2)CCC(N=[N+]=[N-])C1 C(=O)(C1=NOC(C)C1)NCCN1CCN(C(c2c(C)sc(O)n2)=O)CC1 N1(C(Cc2nc(C)[nH]n2)=O)CCCC(CCCCNC(=O)Cc2cnccn2)C1 C1(O)(CC#C)CCN(C(C2(CNC(=O)CC3CCC(O)C3)CCCO2)=O)CC1 N1(C(C(C)OCC#C)=O)CCN(C(c2ccc(CC)c(F)c2)=O)C(C2CC2)C1 C1(C(NOCCC)=O)CC(C)CCN1C(C1CC=C(C)CC1)=O C1(C(=O)NCc2c(C)n[nH]c2C)CCC2C(C1)C2(F)F.C1(OC)CC(CO)C1OC C(=O)(C#CC1(CC)COC1)NC(CNC(COCCCOC)=O)CC c1(C(=O)NC2CC3CC(NC(C(C(C)C)OC)=O)C3C2)ccc(F)c(C)c1C#N N1(C(Cc2scc(C)c2)=O)CCC2(CCN(C(=O)C(C)C3CCOC3)C2)C1 N1(C(c2nccc(SC)n2)=O)CC2CC(Nc3cc(O)nc(O)n3)CC1C2 c1(C(=O)NC(C(C)NC(c2cnn(C(C)C)c2F)=O)CO)cc(F)ncc1OC N1(C(c2c(C)nc[nH]2)=O)CC(C(=O)NC2C(C)C2(C)C)C(C)(C)C1 C(C(=O)N1CCCC1(C)CCC(=O)NC(C(C)(C)O)C1CC1)(C(C)C)SCC Oc1cc(-n2nc(-c3ccncc3)nc2C2CCCC(O)C2)ccn1 C1(N(C(C(C)c2ccco2)=O)CCO)CCN(C(=O)CCCc2ncco2)C1 C1(CN(C(CCc2c(C)n[nH]c2)=O)C)CN(C(=O)CCCC2CC2)CC12CC2 c1(C(=O)NC)cccc(NC(=O)CCC2CCN(C(c3cc(C)[nH]n3)=O)C2)c1 C1(NC(C2(CNC(C3C(C)(C)OCC3)=O)CC23CCC3)=O)Cc2cscc2C1 O=C(O)C(n1ccccc1=O)N1CCCC1C=Cc1ccccc1 N1(C(C(CC)(C)C)=O)CCN(C2CCOCC2)C(C)C1 O=C1CC(NC(c2ccc(-c3cn(-c4ccncc4)nn3)s2)=O)CCN1 N1(C(COCCC(C)C)=O)CC2CC(NC(C3CC4(C3)CC(C)C4)=O)C1C2 c1(C(=O)NC2CN(C(=O)CC3(O)CCCCCC3)C2)cccc2[nH]nc(O)c12 Cc1cnc(CC(=O)NCC2CC(NC(=O)C=C3CCN(C)C3)C2)o1 c1(CN(CCC(N2CC(C)C2(C)C)=O)CC)ccc(C#N)cc1 Oc1c(CC2CN(CCO)CC23CC3)cccc1F c1(C(=O)NC2(CNC(c3occc3Cl)=O)CC2)ccnnc1O Cc1cc(C(N2CCC(CNC(c3ccc(CO)s3)=O)C23CC3)=O)c(O)nn1 CN=c1[nH]c(C(N2CC(NC(=O)CCCNC(N)=O)C(n3cccn3)C2)=O)cs1 C1(C)(C(N(CC(CN(C(=O)Cc2cc[nH]n2)C)O)C)=O)CCC(F)(F)C1 c1(C(=O)NCC2(O)CCCN(C(C(COC)N(C)C)=O)C2)ccn2ccnc2c1 c1(CC(=O)NCCC(C)NC(C2CCO2)=O)c(F)cccc1F C1(CN(C(=O)CC2CCCN2C(c2cc(OC)no2)=O)C)CCCCO1 c1(C(N(CCOCCN(C(C(=O)N(C)C)=O)C)C)=O)c[nH]c(=N)c2[nH]ccc12 c1(CN2CC(C)(C(N3CC(=O)NC(=O)C3)=O)C2)ccc([N+](=O)[O-])c(O)c1 N1(C(c2nc(C3CC=C(C)CC3)sc2)=O)CCN(C(=O)C(C)(C)C)CC1CC#N CC(C)(C)C(CO)C(=O)NC1C=CC(C(N2CC3OCC(CO)C3C2)=O)C1 CN1CCN(C)C(CNC(=O)C(CC(F)F)N(C)C(C2CC=CCC2)=O)C1 C1(NC(C(CC)O)=O)CC12CC(NC(=O)CN(C(=O)C(C)C)C)C2 c1(C(=O)NC2CC3CN(C(C=NOC)=O)C2C3)cc(=O)c2cc(F)ccc2o1 c1(C(=O)NC2CC(NC(C3C(COC)C3)=O)C2)ccc2ccccc2c1F c1(C(N(C(C(=O)NCC2C(C(=O)OC)C2)C)C2CC2)=O)ccncn1 c1(OCC)ccc([N+](=O)[O-])c(C(=O)NCC23CCC(CN(C(C)=O)C2)C3)c1 c1(C(=O)NC2CN(C(COCCC)=O)C2)cc(S(=O)(=O)N2CCCC2)c(C)o1 C(=O)(C1=NOC(C)C1)NC1CN(C(C2(CC)CCNC2=O)=O)CC1C N1(C(CC2CC(CC)C2)=O)CC2CCC1CC2NC(c1cnn[nH]1)=O C(=O)(C(C)(C)CCCF)NC1CC(C)(NC(CCc2cc(C)n(C)n2)=O)C1 N1(C(C2(COC)CCCCC2)=O)CC2CC(C1)N(c1cc(C)nc(COC)n1)C2 N1(C(c2cnn(C)c2N)=O)CC2(C1)CN(C(C1CC1(C)C(F)(F)F)=O)CCO2 c1(C(N2CCC(NC(Cc3cc(C)on3)=O)(CF)C2)=O)ncnc(O)c1Br CC1CC(C(=O)N2CCC(NC(c3c(C(F)F)cnn3C)=O)C2)=NO1 c1(C(=O)NCC(C2N(C(C=CC(CC)=CC)=O)CCC2)(C)C)ccc(C)c(O)n1 C(=O)(C1=C(C)CCCC1(C)C)NCC(C(C)(C)C)NC(CC(CC)(C)C)=O c1(NC(=O)Nc2scc(-c3ccc(CC)cc3)n2)cc(Br)ccc1OC n1(CC)nc(C)cc1C(=O)NC1CCCC(NC(C2CC(C(F)(F)F)C2)=O)C1 C1(C(=O)NC(C)CCNC(C2(C)CSC2)=O)CCc2cnn(C)c2C1 c1(CCC(=O)N(CC(CNC(C2C(CCOC)C2)=O)C)C)cccn1C N1(C(C2CCN(C(C(C(C)C)OC)=O)CC2(C)C)=O)CCC2(C=CCO2)CC1 C(=O)(C(F)CCC(C)C)NCC(CCOC)NC(c1ccncc1N)=O c1(C(C)CC(=O)NC2(C(=O)O)CCC2C(=O)O)ccc(F)cc1F O(NC(=O)CCC1(NC(=O)Cn2cnnc2)CCC1)CC(C)(C)O Cc1cc(C(=O)NCC2(O)CCN(C(C3(C4CCCO4)CC3)=O)C2)n(C(F)F)n1 CCC(Cc1nc(-c2ccc(Cl)nc2)nn1Cc1cc(C)nc(C)c1)CC(F)F C1(CNC(CCNC(C)=O)=O)CN(C(=O)C(C)c2ccsc2)CC1C CC12CCOC(C(N3CCC(NC(c4ocnc4C4CC4)=O)C3(C)C)=O)(C1)C2 N1(C(c2cc3cccnn3c2)=O)CCC2CCN(c3cc(F)ncn3)CC2C1 c1(C(N2CCCC(C)(C(=O)Nc3c(C)cc(Cl)nc3)C2)=O)onc2ccccc12 C(=O)(CCCC(C)(F)F)NC(CNC(COC(C)C)=O)C(C)C(C)C c1(C(NNC(c2c(C(=O)OC)nn(C)n2)=O)=O)cccc2cnccc12 C1(OC)CC2CN(C(=O)C(c3cncnc3)C)Cc3cccnc3N2C1 C(CCC)(C(=O)N1CCC(C)(NC(c2cc(OC)no2)=O)C1)=CCC C1(O)(Cc2onc(CN(C)OCC)n2)CCCN(C(=O)C(C)(C)CF)C1 C(=O)(C(CC(=O)OC)N(C)C)NCCCCNC(C(CCC)O)=O c1(OC)ncc(C(=O)O)cc1C(=O)NCC(c1ccc(C(F)(F)F)cc1)(F)F c1(N2C3CCC(NC(C(C(C)C)NC(C)=O)=O)C(C3)C2)ccc([N+](=O)[O-])c(O)n1 CC(C)C(F)C(=O)N(C)CC1(C)CCCC1NC(c1ccc(F)s1)=O C(c1ccnn1C)=CC(=O)N(CCCC(=O)NCCc1scc(C)n1)C N1(C(c2c(C)c(F)cnc2)=O)CC(C)N(C(=O)C(C)C(C)C)C(C)C1 N1(C(c2c(C)[nH]cc2)=O)CCC2CCCC12CNC(c1cn(C)c(C)cc1=O)=O c1(N(C(=O)NC(C(C(=O)OC)C)C)C2CC2)cc([N+](=O)[O-])ccc1C(F)(F)F C[S+](C)CCC(O)C(=O)N1CC(Cn2cc(-c3ccccc3OC(F)F)nn2)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CC(C(=O)NC2CCNC(=O)C2)CC(C)(C)C1 C1(CNC(=O)CC2(COC)CC2)C2CN(C(=O)CC3CCCN3C)CC12.C(=O)OC N1(C(Cn2cc(CNC(C(C(=O)OC)OC)=O)nn2)=O)CC2CC3CC2C1C3O N1(C(c2nc(OCC)oc2)=O)CCN(C(=O)CC2CC(OC)C2)CC1CC CC1CN(C(=O)CN2CCN(C)CC2)CCC1NC(=O)CC(C)(C)c1cccs1 C(C)(CO)(C(=O)NCc1nc(CO)ns1)NC(CNC(C1C(C)C1)=O)=O N1(C(=O)CCF)CC2CC(C1)N(C(=O)C(Cc1ccccc1)C1CCCC1)C2 N1(CCC(=O)NC(C(C)NC(c2cn(C)c(O)n2)=O)C)CCc2ccccc2C1 C1(NC(C(CN(C(CCCCSC)=O)C)C)=O)C(O)C2CCCC12 C(=O)(CCC(=O)NC1CC(NC(=O)CC(O)C2CCCC2)CC1O)OC(C)(C)C N1(C(c2c(C)snc2)=O)CCC2(CC1)CC2(CO)CNC(=O)CCCC1CCC1 c1(CC(=O)NCCCC(C)NC(CC2ON=C(C)C2)=O)cccc(F)c1O c1(OC)c(C)cc(CC(N2CCOCC2CNCc2ccc(F)nc2)=O)cc1C C1(C(=O)NCC2(O)C(C)CCC2)CN(C(=O)C=CC(=O)NC2CC2)CCC1(C)C c1(C(=O)OC)n[nH]c2c1CN(C(c1c(F)cc(Cl)cc1Cl)=O)C2 C1(CC(=O)NCC(C)CNC(C2CC(N(C)C)C2)=O)CCC2(CCC2)O1 c1(C(=O)NC2CCCN(C(CC3OCC(C)(C)OC3)=O)C2)ccnc2c1CCO2 c1(CN(C)Cc2cccc(C)c2)cc(Cl)c(Cl)n1C c1(C(N2CCC2c2cn(CC(=O)O)nn2)C)cnn2c1OCC(C)(C)C2 Cn1cc(NC(C2CC(CC(=O)NCC34CCC3C4)C2)=O)c(OCC(F)F)n1 C(CN=c1[nH]c2ccc(O)cc2s1)NC(c1cccc(=S)n1O)=O.c12ccccc1S2 N1(C(c2cn(CC)nc2)C(=O)NCC2CC2)CCC(C)C2(CCC2)C1 c1(C(C(=O)N(CCNC(C(C)SCCCC)=O)C)OC)ccccc1F C1(=O)C(C)(C)C2=CCN(C2)C(=O)N1.Cc1cnc(Br)cc1C(=O)O C1(NC(C2CC(C(C)C)C2)=O)C2CC(NC(=O)C(F)(F)CO)CC12 C1(C(=O)NCC2(SC3CC3)CCC2)CCN(CC(F)F)C1 C1(NC(C2(C#C)CC2)=O)CC(CNC(c2ccc(C(F)(F)F)[nH]2)=O)C1(C)C CN1CCC(C(N2CCC(C(O)CNC(c3cc(C(N)=O)no3)=O)CC2)=O)C1=O C1(C)(C(C)C)CN(C(C2CC(NC(c3ccc(C#N)s3)=O)C2(C)C)=O)CCO1 C(=O)(CC1C(=O)N(C)c2ccccc21)N(CCC)CCNC(C1OCCOC1C)=O C1(C(=O)NC2(C(=O)NCCSC(F)F)C(C)C2)CN(C)CCN1C Cc1cc2[nH]c(C(=O)NCC(C)(C)CN(C(=O)C(C)N3CC(C)C3)C)cc2o1 c1(OCCOC)cncc(C(=O)NCC(C)(O)CNC(=O)CC2(C3CC3)CC2)c1 c1(CNC(C2(C)CCC(OCC)CC2)=O)cnn2c1CN(c1cnsn1)CC2 c1(NC(CC)=O)cccc(NC(=O)C#CC2CC2)c1 c1(C(=O)NCC2N(C(C3C(C=C)CC3)=O)CCC(C)C2)cc(=O)c(OC)cn1C c1(C(c2n(CCCCCC)nnn2)NCc2cnoc2)c(C)nn(C)c1C(F)F N1(C(C(C)NC(C(C)SC)=O)=O)CCC(C(C)(O)CNC(=O)COC(C)C)CC1 c1(C(C(=O)NC2(C)CCN(C(C(C)C(F)F)=O)C2)=O)cc(Cl)cc(Cl)c1 c1(N(C)CCC2CCOC2)ccncc1S(=O)(=O)N1CCOC(CS(C)(=O)=O)C1 c1(CNC(C(c2cccc(C#N)n2)N(C2(C#C)CC2)C)=O)ccc(F)c(Cl)c1F c1(CC(=O)NC2C(CNC(C(CCC)OC)=O)CC2)ccc(C)cc1Br N1(C(COCCOCC#C)=O)CC(C(=O)NCC(CC)CO)(CC)C1 c1(CNC(CCc2ccc(C)s2)=O)ccc(CNC(=O)CC2CCOC2C)cc1 N1(C(C2(CCC=C)CN(C(c3ncncc3C)=O)C2)=O)CCOC2CCCC12 C1(COC)(CNC(C2CNC(=O)N2)=O)CCCN1C(=O)CCc1ccccc1 N1(C(CCOC(C)C)=O)CCOC(C(=O)NCc2cc(C(=O)C3CC3)n[nH]2)C1 Cc1cc(F)ccc1N(C)C(=O)N(C1CC1)CC1(c2ccc(Br)cc2)CCCC1 C1(C(=O)NCc2onc(CCC)n2)COCCC1C C1(C(=O)NC(C2CCCC2)CNC(CSCC#C)=O)CC12CC(=C)C2 CC1CCN(C(C2CC(O)CCN2C(c2cnnc(O)c2)=O)=O)C1(C)C C1(CNC(c2c(C)nc(CCC)s2)=O)CN(C(C2CCCCO2)=O)CCN1C c1(OCC)ccc(N)c(C(=O)N(CC(C)CNC(c2cscc2Cl)=O)C)c1 C1(NC(C2(OCC)CCCCC2)=O)CCN(C(=O)CCC2CC2(C)C)CC1O N1(C(CCCC(=O)OCC)=O)CCC(C2(NC(c3ncccc3SC)=O)CC2)C1 Cc1cc(=NC(Cc2ccccc2)NCc2ccc(F)cc2Br)c([N+](=O)[O-])c[nH]1 C1(C)(C(=O)NC(C)C=CC(=O)NCCC#CCO)CCCCC1C c1(CC(C)C(=O)NCCn2ccnc2)ccc(Br)cc1 CC1(C)COC(CC(N2CC(OCCNC(c3cncc(Cl)c3)=O)C2)=O)CO1 N1(C(CSCC=C)=O)CCOC(c2cc(NCC3CC3)c(O)nn2)C1 C1(NC(=O)C(C2CCCO2)C2CC2)CC2CN(C(=O)C=C3CCCCC3)CC12 c1(CCCCC)ccc(SC)cc1.C12CCCC(C1)OC(=O)CO2 c1(C(N(CCC(=O)NC2CCC2C)CC=C)=O)cn(C)c(C)n1 C(=O)(C#CC1CCCO1)N(C1CCCCN(C(c2[nH]nc(CC)c2Cl)=O)C1)C N1(C(C2(CNC(=O)CC3C=CCCC3)CC(=C)C2)=O)CCC(F)(F)C(F)C1 CN1C(=O)CCC1C(=O)NCC(C1CCCN1c1nc(C(C)(C)C)ns1)(C)C C1(CN(C2CCC(n3cc(C4(C=O)CCCO4)nn3)CC2)C(CCC(C)O)=O)CCOC(C)(C)C1 N1(C(CNC=O)=O)CC2(CC(CNC(c3ccc(F)c(C(F)F)c3)=O)C2)C1 C1(C(N2CC(CSC)C2)=O)CC2(CCN1C(c1cncc(Cl)c1)=O)CC2 c1(C(=O)OCc2cccc(SCC)c2)ccc(Cl)c(Br)c1 c1(CNC(=O)C(=O)NCCc2csc(CNC3CCC(F)C3)n2)ccc(F)cc1 c1(-c2ccc(SCC)o2)cn(CC)[nH]c1=N.C(=O)(C(F)C(C)C)NC.N12CC(C1)C2=O N1(C(c2ccc(OC)cc2)=O)CCC2(CC1)CC2CNC(C1(C)CNC(=O)C1)=O C(=O)(CCCCC(C)(C)OC)N1CCCC(O)(CCNC(C(CC)O)=O)C1 c1(CC)ccc(C(=O)NCC23CC2CN(C(=O)CC(C)n2ccc(C)n2)C3)cn1 CC(C)C(C(=O)N1CCCC(CCNC(=O)Cc2ccccc2F)C1)NC(N)=O C=C(Cl)CC(C(=O)N1CCOC(C)C1CO)NC(C1CC1C1CC1)=O c1(OC)cc(C(N2CCC(C)(NC(c3ccccc3F)=O)CC2)=O)cc(F)c1F O=C(C1=NOC(CO)C1)N1C(CNC(c2ncoc2C2CCC2)=O)CC1 c1(C(=O)NC2CN(C(=O)CCN3CCCCC3=O)C2)cc(F)cc2nccnc12 c1(C(N2CCC(NC(C(C)c3cccs3)=O)C2)=O)ccncc1C(F)(F)F c1(C(C)CC(N2CC3CC2C3NC(=O)CN2CCNC2=O)=O)ccc(F)cc1F C1(C(=O)NC2(CC(=O)NCc3cccnc3F)CCC2)Cc2nccn2C1 n1(C(C(=O)NCCN(CCOC)C(C2CCOC2)=O)C)cc(C)cn1 C1(CNC(CCCCOC)=O)(NC(=O)C(C)c2cccs2)CC2CCC1CC2 CC1CC(CNC(=O)C(C)Cc2ccnn2C)CN(C(C23CC4CC2C3C4)=O)C1 C(C1=CCCN(C)C1)NC(CCCC1(NC(C(C(C)C)OC)=O)CCC1)=O N1(C(C2CC(CC)(CC)C2)=O)CCN(C)CC1CN(C(=O)C1=CCCCO1)CC CCCCC(CNC(c1csc(COC)n1)=O)NC(c1ccccc1Cl)=O N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CCC1C CC1(C)CNCCN1C(=O)C(=O)Nc1ccccc1N1CCNC1=O N1(C(Cc2cccc(OC)n2)=O)CC2CCN(C(C3CC(SC)C3)=O)CC2C1 N12CC(C3(CC3)C1)n1cc(nn1)C[SH](CC)CC2=O.c1(C(CC)C=O)ccc(Cl)cc1F S(=O)(=O)(c1cc(C)ccc1C)N1CCC2CN(C(C(=C)C(F)(F)F)=O)CC21 C(CC(C)(C)C(=O)NCCc1cc(C(=O)NCC2(CCO)CCC2)no1)OC c1(C(N2CC(CC)C(NC(C3CC(OC)C3)=O)C2)=O)cc(OC)ncc1F c1(C(N2C(CN(C(C3CC3(C)C)=O)CC)CCCC2)=O)cc2cc(Cl)ccc2o1 C1(NC(N2CCCC2CCc2ccccc2)=O)C(O)C(O)CN1 CC(C)(C)C#CC(=O)NCC1(F)CCN(C(=O)CSc2ccccc2)CC1 N1(C(C(C)OCCC#C)=O)CCCC(n2cc(CNC(=O)CCC3CC3)nn2)C1 n1(CC(=O)NCC(C)CN(C(=O)CC2CCCCN2C)C)ccc(=O)n(C)c1=O N1(C(=O)NC2CC(OCC)C23CCOCC3)CCc2ncc(C)n2CC1 C1(NC(C(n2cc(Cl)cn2)C)=O)CCN(C(=O)C#CC2(C(F)(F)F)CC2)CC1C c1(CCCC(=O)NC2C(NC(C(CC)=CC)=O)COCC2)c[nH]c2ccccc12 C12(C(=O)NC(CCN(C(c3cc(COC)cn3C)=O)C)(C)C)CC(C)(C1)OC2C c1(NC2CCCCN(C(C(C=C)(C)O)=O)C2)ncc(S(C)(=O)=O)cc1Cl N1(C(CNC(=O)OCC=C)=O)CCN(C(C2C=CC(CCC)C2)=O)CC1CO C1(C)(CNC(c2n(C)nnc2Br)=O)CN(C(=O)CCn2cnnn2)C(C)(C)C1 C1(C(=O)NC(CN(C(c2cnsn2)=O)CC)C)CCCN(c2cnccn2)C1 C1(CC(=O)NCCN(C)C(c2ccccc2C(=O)NC)=O)Cc2ccccc2O1 C1(NC(=O)CCc2c(F)cccc2Cl)CN(C(=O)CCC2CC2)CC2(CC2)C1 c1(C(=O)NCC2CCC(C)N(C(=O)CCCF)C2)cc2c(nn1)CCCO2 Cc1c(NC(C2CC(=O)CN2C(=O)C(C)(O)CN(C)C)=O)cccc1C#N c1(C(C(=O)NCC2CCCN2C(C2COC2)=O)O)ccc(Cl)cc1 c1(C(=O)NCC#CCNC(CC(=C)Br)=O)c(C)noc1C(F)F c1(C(N2CCC(CNC(CCCOC)=O)(OC)C2)=O)cnc2n1C(C)CCC2 C1(SC(C(=O)NCCCC)CC)CNCC1(C)C CC1(C)CC(=O)NCC1C(N1CCN(C(c2c[nH]nc2F)=O)CC1CC(F)F)=O c1(C(C)(C)C)ccc(C(=O)NC2CCC2NC(c2ccccc2)=O)[nH]1 c1(C(N2CC3C(NC(C4CC(=O)NCC4)=O)C3C2)=O)ccc2c(c1)COC2 CC1CC=C(C(=O)N2CC(C(=O)NC3CC(CCC(N)=O)C3)C(F)C2)CC1 c1(CC)ccc(C(N2CCC(CN(C)C(C3CN(C(N)=O)C3)=O)C2)=O)cc1 N1(CC(CNC(=O)Nc2snc(CC)n2)O)CCN(C)CC1 N1(C(=O)CCOc2ccc(Br)cc2)CCCN(C(=O)CO)CCC1 N1(C(C)=O)C(C(=O)NCC(F)(F)C2CC2)CC2CCCCC12 C(CC(C)C(=O)N1CC(OC)CC1C(=O)NC(c1nccc(C)n1)C)OC Cc1cc(CNC(=O)C(CO)NC(c2cccn2C)=O)nn1C C1(CC)CCCC1(C)C(=O)NCC(C)CN(C)C(c1cnc(C(F)(F)F)nc1)=O C#CC1(C(=O)NCC(C)CNC(=O)CCC2(C)CC2(F)F)CCCC1 c1(C(=O)NCC=CCNC(Cc2nc(C)sc2C)=O)ccnc(O)c1Br c1(=O)nc2nc(s1)NN2.c1(C(N(C)C)=O)cccc(C(N2CCCC2C2CC2)=O)c1 C1(N)CCC12CCNCC2.Cc1nc(C2CC2)sc1CC(C(=O)CCCC#N)=O C1(C(=O)NCC2(CNC(C3CCC(NC(C)=O)C3)=O)CC2)NC(=O)CC1C C1(C(N(CCN(C(C(C)=CC)=O)C)C)=O)CCN(C2CCS(=O)(=O)C2)CC1 c1(CN2CCC(C)(NCc3cc(Br)no3)C2)ccc(-n2cccn2)c(F)c1 N1(C(c2c(CC)oc(C)c2)=O)C2CCC1CN(C(=O)C(C)(C)Cn1cncn1)C2 CC1(C)COCC(C(=O)NC2CC2NC(c2sccc2F)=O)O1 c1(C(=O)NCC2CC(NC(C3CS(=O)(=O)N3)=O)C2)coc2ccc(Cl)cc12 C=CCCC(C(=O)OC)NC(C1CC1c1cccc(F)c1)=O c1(CC(=O)NC2CN(C(=O)CCc3ccccc3)C3CC23)ccnc(C(F)(F)F)c1 C1(NC(=O)OC(C)(C)C)CC2(CCN(N3CC(OCC4CCC4)C3)C2)C1 Cc1ccc(Cl)c(OCC(=O)NCCCCNC(c2csc(S)n2)=O)c1 C=CC1CCN(C(C2CCCC2CNC(c2conc2C)=O)=O)CC1 N1(CC(N2CC=CC2CNC(C2(Br)CC2)=O)=O)CCCCC(O)C1=O C1(C(=O)NC2CCC(CNC(C3CCC(=O)N3C)=O)C2)(CC)CCOCC1 C1(C(N2C(C)CCC2)=O)CC2CC1CC2NC(c1ccc(F)cc1)=O c1(CNC(C2CCC(=O)NC2)=O)cnn2c1CN(Cc1ccc(O)cc1Cl)CC2 c1(C(=O)NC2C(CO)CCN(C(C=CSC)=O)C2)[nH]nc2c1CCCC2(C)C c1(CC(=O)NCCC(CC)(C)NC(=O)C(F)C(F)(F)F)ccc(C)cc1C CN1CCN(C(=O)CC2(C(F)(F)F)CC2)C(CNC(=O)CN2CCOC2=O)C1 Cc1coc(C=CC(N2CCN(C(C3CC(C)C3)=O)CC2)=O)n1 C1(COC)(NC(=O)C=C2CCC2)CCN(C(c2ncccc2CC2CCC2)=O)C1 c1(CSCC(=O)NC2(CNC(c3c(C)cccc3O)=O)CC2)ccc2c(c1)OCO2 CCCCCCN(CCCN(C(=O)C(c1cnn(C)c1)O)C)C N1(C(C(C)CN(C)C)=O)CC(C(=O)NC2CC=CCC2)CC12CCC2 N1(C(C(CC(=C)C)OC)=O)CCC2(CCCC2NC(c2nc(Cl)cs2)=O)CC1 Cc1cccc2oc(C(=O)N(C3CCN(CC(C)CC(C)C)C3)C)cc12 C1(CNC(C(CC)Oc2ccccc2Cl)=O)(CO)CCCN(C(=O)CC(C)C)C1 S(=O)(=O)(c1ccccc1Br)NC(C(=O)NCCCCCC)C(C)O Cc1nn(C)c(F)c1C(=O)NCC1CCCCN1C(=O)CC1COCC1O C12(CNC(=O)C=CBr)CN(C(=O)Cn3ccccc3=O)CC1CCO2 N1(C(c2cc(OC)n[nH]2)=O)CCC(CF)(NC(=O)COC2CCN(C)CC2)C1 N1(C(C(C)O)=O)CC2CC(NC(=O)COc3ccc(F)cc3Br)CC(C2)C1 Cc1ccnc2nc(C(=O)NC(C)C(C)(C)NC(=O)CN3C(C)CCC3C)nn12 C(=O)(CC1=CCN(C(c2ccc(C)cc2C)=O)CC1)N(C1(C(=O)OC)CC1)C C1(C(N(CC(=O)NC(c2c(C)ncs2)C)CC(C)C)=O)CCCCC(=O)N1 c1(OC)cc(F)c(NC(N2CCOCCC2C2CC2)=O)cc1OC S(=O)(=O)(c1cccc(=NCCn2cncn2)[nH]1)N1C(CNC(N)=O)CCC1 c1(CC(=O)NC2CC(NC(C3(O)CCOC3)=O)C2)cscc1Br CCC(O)(CNC(=O)C(C)N(C(c1cnn(C)c1OC)=O)C1CC1)CC N1(C(c2ccc(COC)o2)=O)CC(NC(=O)CC2CCOCC2)C(C)C1 c1(C(=O)OCc2nccc(OC)n2)cc(F)cc2c1NCCC2 S(=O)(=O)(c1cnccc1N1CCC2(C1)OCCO2)NCc1ncc(C)nc1 Cc1nc(C2CC2)sc1C(=O)N(CCCNC(=O)CSC(F)F)CCO C1(NC(CC2CC(SC)C2)=O)CN(C(C2CC(=O)CCO2)=O)CC1(C)C C(=O)(C(COC)NC(=O)CC(C)n1cccn1)OC.C12CC1C(C)NC2=O C1(NC(COCCOCC#C)=O)CN(C(=O)COCC(F)(F)F)CC(C(F)(F)F)O1 C(C(=O)N=c1ccn(C(F)F)[nH]1)(C1CCC1)NC(c1ccc(C2CC2)o1)=O N1(C(C2(CC)CCCO2)=O)CC2(CCCC(CNC(c3ccc(Cl)cc3)=O)O2)C1 CC(C)C(CNC(=O)COCC1CC1)NC(=O)C(c1ccccc1)O c1(C(N2C(C)CC(F)C2)C(=O)NCC2CCS(=O)(=O)C2)cccc(C#N)c1 N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CC=CCC2)C1 C1(NC(c2n(C)cnc2)=O)CC12CC(NC(C1COCC1C(F)F)=O)C2 C1(NC(c2ccc(C)nc2)=O)CC2CN(C(c3cnco3)=O)CCN2C1=O c1(C(=O)NCC2CCC(NC(C(C(C)C)N(C)C)=O)C2)ccc(=O)n(O)c1 C1(NC(C2C(C(C)C)OCC2)=O)CC=CCC1C(N1CCCCC1CCO)=O C(C(C)C(C)C(=O)NCC1=CCN(C(c2cc(O)nc(OC)n2)=O)CC1)OC N1(Cc2c(C)n[nH]c2C)CCC2(CC1)C(O)CC(C(=O)O)C2 C1(C(=O)NCC2CN(C(C)C)C2)CCC(C2CC2)N1C(=O)C=Cc1cc[nH]n1 Cc1ccc(N2CC(C(=O)NCC3CCN(C)C3)CC2=O)cc1C C(=O)(C(F)CCC(C)(C)C)N(CCN(C(c1cn(CC=C)nc1)=O)CC)CC N1(C(C(F)=CC)=O)CC(C)(C)OCC1CNC(=O)COc1cc(F)ccc1F N1(C(C(C)CC(N)=O)=O)CC(NC(=O)CS(=O)(=O)N(C)C)CC12CCCCC2 CC1CN(C(c2cc(Br)cc(N)c2Cl)=O)CC(C)C1NC(=O)C=CC1CC1 O=C(CCCC(F)C(=O)O)N1CCC(F)(c2ccccn2)CC1 c1(C(N)=O)cccc2c1CN(C(=O)CC1CCN(C(C3CCC(=O)O3)=O)CC1)C2 CCC(C)CC(C)C(=O)N1CCC(C)(C)C(NC(=O)Cc2cc(C)ccc2F)C1 C1(CNC(C(C)O)=O)CCC2(CN(C(c3ccc(F)cc3O)=O)C2)O1 C12(C(=O)NC3(CO)CN(C(CC(CC)C)=O)C3)CCC(CO)(CC1)CC2 c1(C(N(CC(CNC(c2cnc(OCC)s2)=O)C)C)=O)nc(O)nc(O)c1N N1(C(C(N)=O)=O)CC2(CCN(C(=O)CNC(c3ccc(Cl)c(N(C)C)c3)=O)C2)C1 N1(C(C2(C)CC2C(F)(F)F)=O)CCCC1(C)C(=O)NCC1CCCOC1 C1(NC(NCC(C(C)(F)F)(C)C)=NCc2ccsc2)CCOC2(C1)CS(=O)(=O)C2 c1(CNC(C(COCC)NC(C2CCSC2)=O)=O)ccccc1CO C1(CNC(C(C)NC(C)=O)=O)CN(C(C2CC2C2(C)COC2)=O)CCC12CCC2 C1(C(N2CC(CC(=O)N(CC(C)(C)OC)C)OCC2)=O)CCC(O)CN1C c1(CNC(C23N(C(c4cnn(C)c4Cl)=O)CC(C2)C3)=O)c[nH]c2ncccc12 c1(C(=O)NC2C(NC(c3ccn(CCOCC)n3)=O)CC2)cc2c[nH]cnc-2n1 c1(C(=O)NC(C(C)NC(c2nnc(CC)s2)=O)(C)C)ccn2c(C)ncc2c1 N1(c2cc(NC3CCC(C=O)O3)ncn2)CCOCC2(CCC2)CC1.CC(C)C c1(C(N2CCCC(CN(C(C3C(C#C)C3)=O)C)C2)=O)cc(Br)c(F)cc1N CC1(C)CN(C(=O)CCNC(C2CCC2)=O)CC(CNC(c2ccc(F)o2)=O)O1 CCC(COC)C(=O)NCC(CC(=O)NC(C)(CO)CO)C1CCC1 N1(S(C(CCC)CC)(=O)=O)CCOC2(CCSCC2)CC1 CCS(=O)(=O)NC(C)C(=O)N(CC(C)(C)NC(=O)C(C)c1ccco1)C C1(NC(c2n(CC)nc(C(C)C)c2)=O)CCCN(C(=O)C2=CCCO2)CC1 Cn1cnn(CC(N2CCC(C(O)CNC(=O)C(O)C3CCC3)CC2)=O)c1=O c1(CC)nn(C)c(CC)c1NC(=O)Nc1cccc(-n2ccnc2O)c1 C(C1CCOc2ccc(Br)cc21)NC(c1n[nH]c(C)c1F)=O c1(C(=O)NCC(C)(CO)NC(C2CC3CC3C2)=O)nc2n(c1Cl)CCCC2 C12(CNC(C(CC)(C)C)=O)CN(C(c3sccc3S(N)(=O)=O)=O)CC1CCO2 Cc1cc(C)c(C(=O)NCC2=CCN(C(C3(C#N)CC3)=O)CC2)c(S)n1 N1(C(C(C)CC2CC2)=O)CC2(CC(CNC(=O)Cn3cnnn3)C2)C1 C1(NC(CCCOCCC)=O)CC(NC(c2cnn3c2CCC3)=O)C12CCC2 C1(N(C(C2C(=C)C2)=O)CC)CCN(C(=O)C=Cc2ncc[nH]2)CC1 N1(C(c2c(CN(C)C)cco2)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC1CF CC1CC(F)(F)CN1C(C1CSCCN1C(=O)C=CC(F)F)=O Cc1cc(C(N2CCC(NC(=O)COCC3CCCO3)C(F)C2)=O)c(C)cc1Cl c1(OC)cc(C(=O)OCCOCCN)cc([N+](=O)[O-])c1OC.C(C)(C)(C)O C1(C(N2CCN(C(CC)=O)C(CC)C2)=O)CC2CC1CC2(F)F C1(CC)(N)CCN(C(=O)CC(O)CNC(=O)OC(C)(C)C)CC1.C(=O)(CCF)NC c1(C(=O)NC(CCC(=O)O)CCCCCC)cc2cn[nH]c2cn1.NC CCC(C(=O)N1CCC(NC(c2sc(C3CC3)nc2C)=O)C1)C(C)(C)CC c1(C(=O)NC2CC2C(N2CCS(=O)CC2)=O)cc(O)nc(O)c1 C12(C(=O)NCC(COC)C)C(NC(=O)Cc3nonc3C)C3CC1C2C3 C(=O)(CCCCCNC(C1CC2COCC2C1)=O)N(CC(COC)O)C N1(C(Cc2ccc(C#C)cc2)=O)CCN(C(=O)CSCC)C2COCC12 CC(C)(F)CCC(=O)NC1CCOC(C(N2CCC3C(O)CC23)=O)C1 CC(C)CCCCC(C)NC(c1nnnn1C)C1CC1C(C)C c1(C(=O)NCC2CN(C(CCc3onc(C)n3)=O)C2)cc(F)cnc1Cl C1(NC(CC2ON=C(C)C2)=O)CCN(C(C2CCCN2C=O)=O)CC1 C1(CC)CN(C(=O)C=Cc2cccc(OC)c2)CCC1NC(=O)Cc1cc[nH]c1 C12(NC(C(CC)OC)=O)COC(CNC(c3c[nH]nc3-c3ccncc3)=O)(C1)C2 N1(C(C(CC)CC2CCCC2)=O)CC(NC(c2ccon2)=O)CC12CCOCC2 C1(C)(C(N(C(C=C)C2CC2)C)=O)C=CCN1C(C1OCCC1(C)C)=O C1(C(=O)NC2CC(N(C(C=Cc3n(CC)ncc3)=O)C)C2)CN(CP(C)(C)=O)C1 C1(NC(C2C(C(C)NC(C(C)=C(C)C)=O)C2)=O)C(O)CC1O CCCCCC(=O)N1CCN(C2CCN(C(=O)C(C)OCCCC)C2)CC1 c1(-c2c(C)c(F)ccc2)cnn2c1CN(Cc1ccccc1C#N)CC2 C1(CC(=O)NC2CCC(C)(CNC(c3cnc(C(F)F)s3)=O)C2)CCC2(CCC2)O1 C(CC(=O)N(C)Cc1ccc[nH]1)N(CC=C)C(C1CSC1)=O C(CC(C)(C)CC(=O)NC(CCN(C)C)C(=O)N1CC(OCCF)C1)OC Cc1cnc2[nH]cc(CCNC(C3(CNC(=O)CC4CCC4)CC3)=O)c2c1 CC1CN(C(C2CCCN2N=O)=O)CC1(C)CNC(=O)CC12CCCN1CCC2 C1(CNC(CNC(C2CC2Cl)=O)=O)(CO)CC=CC1 Cc1cnncc1C(=O)NCCC1CSCCN1C(c1cc(Cl)cn1C)=O C1(C(=O)NC(CNC(c2c(CC)nc(C)o2)=O)CO)CC2(CO1)CC(F)(F)C2 n1(CC(=O)NC2CN(C(C3ON=C(C)C3)=O)CC(O)C2)c([N+](=O)[O-])cnc1C Cc1c(C(NC2CCCn3nccc32)=O)oc2ccc(I)cc12 c1(C(=O)NCCCCCN(C)C)ccccc1-n1cc(-c2cccc(Br)c2)nn1 C1(C)(C(=O)NCC#CC(=O)NCCCCOC(C)C)CCCOC1 C1(=O)C(CCC2CC2)N1.C1(C(C)C)(NC(=O)CSCC(F)F)CCC1 N1(C(c2nc(OCC)sn2)=O)CCC(NC(=O)CC(C)(F)F)CC1C N1(C(CCc2scc(C)c2)=O)CCC(NC(c2cnc(O)n2C)=O)C(O)C1 CC(F)(F)C(C)(C)CC(=O)N1CCC2(CCCN2C(=O)CCSC2CCCC2)C1 N1(C(CC(COC)NC(=O)C(F)C(C)C)=O)CC2COCC2(C)C1 c1(CNC(=O)COc2ccsn2)cc([N+](=O)[O-])ccc1N1CCCC(C)(CO)C1 C(=O)(C(O)C1=CCCCC1)NC(C)C(C)C(=O)N(CCCCO)C c1(NC(=O)OC(C)(C)C)ccc(C(=O)Nc2ccn(C3CCCCO3)n2)cc1I C12(NC(C(C)C(C)O)=O)CCC(CNC(=O)CC3CC4(CC4)CO3)(C1)OC2 C(=O)(C(F)C(=O)NC(C)C(CO)NC(c1cnn(CC(F)F)n1)=O)OCC CCC(C)C(O)CC(=O)N1CC2CC1C2CNC(=O)C=C=C(C)C S(=O)(=O)(c1ccc(NC)c(C#N)c1)N1CC(C)CC(NC(CC(=O)NC)SC)C1 N1(C(C(C(CC)C)N(C)C(c2cnn(C)c2)=O)=O)CCCN(CC)C(=O)C1 Cc1cc(C(=O)NC23COC(CNC(C4(C)CCC4)=O)(C2)C3)c(C)cc1Cl C1(C2CN(C(C3CCCSC3)=O)C2)(Nc2cc(OCC)ncn2)CC1 N1(C(C2CC(CC)N(C(c3cc(C)nc(C)n3)=O)CC2)=O)CCC12CCCSC2 c1(C(N2CC3CC(NC(C(=O)NC4CC4)=O)C3C2)=O)cnc2c(c1)CCCC2 C1(OC)CCCN(C(=NCCC(=O)Nc2cc(O)nc(C)n2)NC2CC2)C1 CC(CC(N)=O)C(=O)N1CCN(C(=O)CCc2cscn2)C(CO)C1 c1(CC)ccc2[nH]c(C(=O)N(CCCNC(C3(C)CCCO3)=O)CC)c(C)c2c1 C1(NC(c2cccc(C)c2)=O)CCN(C(=O)CC2CCC(C)(C)CO2)CC1C CC(C(F)C(=O)NCC1C=CC(NC(=O)C2=CSCS2)C1)C(F)(F)F c1(C(=O)NCC(N2CC(O)(C(C)NC(c3csnn3)=O)C2)=O)ccc(Cl)cc1 c1(NC(C2CCOC2)CNC(CCNC(c2ccsc2)=O)=O)cc(O)ncn1 C=CCC(C(=O)N1CCC(NC(c2c(C)csc2Cl)=O)CC1C)C(C)C c1(CNC(C2CCCN(C(c3cc(F)ccc3O)=O)CC2)=O)cccc(O)c1F c1(CC(N2CCC(C(CNC(C(CC)O)=O)F)CC2)=O)ccc(O)c(C(C)=O)c1 N1(C(CCCn2cc(C(c3ccccc3)C)nn2)=O)CCC(C)(CO)C1 c1(CCC)n[nH]cc1C(N1CC(C(C(=O)N(CC(C)C)C)NC(C)=O)C1)=O S(=O)(=O)(c1cc(C#N)ccc1Cl)NCc1cccc(CCC#C)c1 c1(C(=O)NC(C2N(C(C3(C=C)CC3)=O)CCCC2)C)ccc(Cl)c(OC)c1 C(=O)(C(C(C)CC)NC(C1CCCN1C(N)=O)=O)NCCOCCC=C c1(CNc2ccc(C(N3C(C(=O)OC)CCCC3)=O)cc2)ccnc(Cl)c1Br N1(C(c2ccc(CC)c(N)c2)=O)CCC(C2CC2)C1CNCc1ncn(CC)n1 C1(C(=O)NCC(c2ccc(F)cc2)OC)CN(C(C)=O)CCO1.C1(O)CCCC1 Cc1cc(C(=O)NCC(O)CNC(=O)C(C)(C)c2cc[nH]n2)c(F)cc1N Cc1c(CNC(=O)C(=O)NCCC2(O)COC2)noc1-c1ccccc1 c1(SC)cc(C(=O)NC(C)C(C)NC(c2ccc[nH]2)=O)ccc1N CCCC(C(=O)NC1CCCN(C(=O)CC=CCc2ccccc2)C1)C(C)C c1(C(=O)NCC(O)COc2cccc(Br)c2)cnn2c1NCCC2 CCC(CC)(CC)C(=O)NC1CCN(C(=O)CC2CC=CCN2C)CCC1CO C1(C(=O)NCCc2ncc(C)o2)N(C(=O)Cc2cnoc2)CCCC1(C)C CC1CN(C(=O)C(C)C(C)O)CC(C)N(C(=O)C=Cc2ccccc2)C1 C1(NC(C(c2ccco2)NC(CC(C)N(C)C)=O)=O)CC2C=CC1C2 C(C)(CC(C)NC(c1cn(-c2ccn(C)n2)cn1)=O)NC(C=C(C)C(C)C)=O C1(C(=O)N(C2CC3CCC2O3)C)(CC)CCCN(C(=O)CN2CCSCC2)C1 c1(C(=O)NC(CC)CNC(c2cc(CO)[nH]n2)=O)oc(C)cc1C C(=O)(C1=NOC2COCC12)N1C(CN=c2snc(C(=O)OC)[nH]2)C(C)CCC1 c1(C(=O)NC(C2CCCCN2C(=O)CCC2CC2(C)C)C)ccc2ccoc2c1 C1(C(=O)CC2C3CN(C(c4cccs4)=O)CC32)Cc2nncn2C1.O=C1CNCO1.N.C Cc1ccc2cc(C(=O)NC(CNC(=O)C(C)(O)C3CCC3)C3CC3)[nH]c2c1 C1(C(N2CCC(C3N(C(=O)Cc4ccco4)CCC3)C2)=O)(C(F)F)CCCCC1 C(=O)(C(=O)N=S(C)(C)=O)NC(C)CC1CCN(C(=O)C2=NOC(CN)C2)CC1 N1(C(CCCOCCC)=O)CC(CNC(c2oc(C3CC3)nc2C)=O)CC1C CC1CC2CCC(C1)N2C(C(=O)NCC1CCCO1)c1ccsc1 C1(C(C(=O)NC2CC(COC)C2)N(c2cnnc(O)c2Cl)C)CN2CCN1CC2C c1(C(N(CCCCCNC(c2n(CC)ncn2)=O)C)=O)ccc(OC)cc1F C1(C(=O)NC2CC(CNC(c3cnc(CC4CC4)s3)=O)C2)CC1C1CCCCC1 Cc1cc(F)cc(C)c1C(N1CCC(C)(NC(c2[nH]ccc2C2CC2)=O)C1)=O c1(OC)ccc(Cl)cc1CC(=O)NCC12CC(CN1C(C1(C)CNC(=O)C1)=O)C2 CN1CC(C)(C)CC1C(N1CCCC1C(C)(C)NC(c1cc2c[nH]nc2s1)=O)=O c1(OC)cc(Cl)c(CNC2CC(C(=O)Nc3ccsc3)C2)c(Cl)c1 c1(Cc2scc(C(S(=O)(=O)NC)C)n2)ccccc1Cc1nn[nH]n1 CCCCCCCNC(C1CN(C(C)C)C1)=O.C12CCN(CC1)C(=O)O2 c1(C(=O)NCCNC(CC2ON=C(CC)C2)=O)n[nH]c2c1COC2 C=CC1CN(C(=O)C(C)O)CC1NC(C1CCOCC1C)=O C1(C(=O)NOc2cccc(Br)c2)CC(C2CC2I)C1 Cc1cn2cc(C(=O)NOCc3cn(C4CCCC4O)nn3)nc2s1 C1(C(=O)NCC2=C(C)CCC2)CCN(C(=O)c2cc(C3CC3)on2)O1 CC12CN(C(CC(=O)NC(c3nc(C4CC4)ncc3Cl)=O)=O)CC(CO)(C1)C2 C1(C(N2CCC(C(C)NC(=O)CC(c3ccccc3)C3CC3)C2)=O)CC2CC1C2 CC1(C)COC(C(=O)NCc2ccccc2CNC(C2CCNC2=O)=O)C1 CC(C)CCCCN(C)C(C1(NC(=O)Cc2ccc(O)nc2)CSC1)=O c1(CNC(C=C)Cc2ccc(F)cc2)cc2n(n1)CCCCO2 N1(C(=O)C2CC2)CCC2(CCCN2C(c2c(Cl)csc2Cl)=O)C1 c12c[nH]c3ccc(cc13)oc2=O.c1(C(CC(=O)OC)C)ccc(OC(C)C)cc1 C1(CC)(NC(c2ncoc2C)=O)CCN(C(c2cnc(O)cc2OC)=O)CC1 CCC(C#N)OC(=O)C(=O)NCCCSC C1(C)(CNC(COC(C)(C)C)=O)CCN(C(=O)CCN2CCCCCC2)CC1 C1(CC(N2CC(C)(OCC)C2)=O)CN(C(C2CCC2)=O)CCO1 N1(CC(=O)NCC(=O)Nc2ccc(C)c(C)c2)CCC2C(C1)NC(=O)N2C n1(CC(=O)NC(C2(O)CN(C(C3C(C)CC=CC3)=O)C2)C)nc2c(n1)CCCC2 c1(CNC=O)ccc(CN)cc1.C1(CCNC(C)=O)COCCOC1.C1C(=O)N1 C1(CC(=O)NCC(C)NC(=O)C=CBr)CC(C)OC1C C1(C2CCN(C(=O)C=Cc3cccs3)C2)(NC(C2CC3CCCCC23)=O)CC1 C1(CC)CCOCCN1C(=O)CCN(C(=O)CCc1cnn[nH]1)CCO c1(SCCC(=O)NC2CN(C(CCCCSC)=O)CC2O)ncnc2[nH]cnc12 N1(C(c2nc(C(C)OC)sc2)=O)CCCC(O)(CNC(=O)CCc2cccs2)C1 C#Cc1cccc(C(=O)NCC2CC2NC(=O)C2=CC(C)(C)C2)c1Cl C=CC(CC)C(=O)NC(C(=O)N(c1cnn(C)c1)CC)C1CCC1 C(=O)(CCC(CF)CF)N1CCC(NC(c2c(OC)n[nH]c2)=O)C1C1CC1 CCC(F)(F)CC(=O)N1CCCN(CCNC(=O)CCC2CCCCO2)CC1 C1(C(C(=O)N(C(C)C)CCN(C)C(C2CN(C)C2)=O)C)CCOCC1 C1(N(CCCC)C(=O)Nc2conc2-c2ccccc2F)CCCCC1C N1(C=O)CCC(CF)C1.C1(CNC(C2(CO)CCO2)=O)CC(C(F)(F)F)C1 c1(C(=O)Nc2c(C)cc(NC(C3(Cl)CC3(F)F)=O)cc2)ccn2ccnc2n1 C(=O)(CC1OCCc2ccccc21)N1C(CNC(c2nc(C)oc2)=O)CC2CC21 Cc1nc(CC(C)C)oc1C(=O)NCCC(C(C)C)NC(C1(CN(C)C)CC1)=O CC1CC(=O)CCC1C(=O)NCC(C1CC1)N(C(=O)CCc1cncnc1O)C c1(C(N2CC(CCNC(CC)=O)OCC2)=O)c(C)cc(OC)cc1F C1(CNC(c2ccc(C(C)=O)[nH]2)=O)COC(C)(C)CN1C(c1cccnc1)=O C1(C(=O)NC2CCN(CCNC(C(CC=CC)C)=O)CC2)CC2C(C1)C2(C)C c1(CC)cc(C)ccc1C(=O)NCCC(C)N(C)C(c1cnc(Cl)c(N)c1)=O Cc1ncc(C=CCNC(C2CCCC2c2ccccc2)=O)s1 c1(C(=O)NC(C2CCN(C(c3ccc(C(C)C)o3)=O)C2)C)ccnc(C2CC2)c1 C1(CC)CCCCC1OCC(=O)NCC1CN(C(C2(CC)CCCO2)=O)C1 C1(NC(C2C(C)CCO2)=O)CN(C(=O)CCc2ccsc2)CC1C1CC1 C1(CNC(=O)CC2CCCCC2)(Cn2cccn2)CCCN1C(=O)CC1CC1 C(=O)(C1=NOC(C)C1)N(CCCNC(c1sc(CC)c(C)c1)=O)CC1CCCC1 CN1C(=O)CCc2ccc(C(=O)NC3CN(C(=O)CC4(O)CC4)C3)cc21 c1(C(CNCCCC)CC)noc(C)c1C(=O)O c1(C(C(C)(C)N(CCc2cn(CC)nn2)C)O)ccc(F)c(F)c1 C1(C(=O)NC(n2cc(Br)cn2)C2CCOC2)C2CC2C2CC12 N1(C(CC2(OC)CC2)=O)CCCC(CO)(NC(C2CCCC(C)(C)C2)=O)C1 c1(C(=O)NCCCN(C(=O)CC2CC(=O)NC(=O)C2)CC)cn2cccnc2n1 N1(C(CCCCCCSC)=O)CC2CCCC(C1)N(C(c1cc[nH]c(=N)c1)=O)C2 c1(C(N2C(C(=O)NCC3(C)OCCO3)CC(OC)C2)=O)ccc2c(c1)CCCC2 C=CCC(C(=O)NC1CCC(CCC(=O)NC(C)C(C)(C)C#N)C1)C(C)C C1(C(=O)NCC2CC(C(=O)NCCCC(=O)OC)C2)Cc2ccccc2C1 C1(CNC(C2C(OCC)CC2)=O)COC(C)(C)CN1C(c1cn(C2CC2)nn1)=O N(C(=NCCC(F)(F)F)NC1COCC1F)Cc1cccc(OC)c1 C1(CCN(C(c2c(CCC)nco2)=O)C)CCCCN1C(c1cnc(C)nc1)=O N1(C(CCc2ncn(C)c2)=O)CCC(O)C1C(N1CC(O)(CC(N)=O)C1)=O C=CCC(C)C(=O)OCc1scc(C(=O)NC(C)Cn2cc(CCCO)nn2)n1 c1(C(=O)NC2C(OC)CN(C(COCC)=O)C2)ccc(Br)c(C)c1F N1(C(CSCCC)=O)CC(CNC(c2c[nH]c(=N)cc2C)=O)C(C)(C)C1 C(=O)(C1CCCc2nccn21)N1CCCC(N(C(=O)C(F)(F)C(F)F)CC)C1 c1(C(N(C)Cc2ccc(CNC(=O)CC(C)(C)F)cc2)=O)cc2n(n1)CCO2 c1(C(N(OC)Cc2ccccc2)=O)cc(S(C)(=O)=O)ccc1NC=O N1(C(C(C)SCCCC)=O)CC(NC(c2cn(CCO)nn2)=O)C(CC)C1 N1(C(c2ccc(C#N)cc2)=O)CC2(CCCC2NC(c2cnsc2)=O)C1 Cc1ccnc(-c2cccc(NC(C3(CC(F)F)CCC3)=O)c2)n1 CCC(CC)(CC)C(=O)NC1CCC(NC(c2oc(C3CC3)nc2C)=O)CC1 Cc1n[nH]c(C)c1SCC(=O)NCC1C2CN(C(=O)CCCn3ccnc3)CC12 C1(CNC(=O)Nc2nccc(P(C)(C)=O)c2)CNCCC12CCOCC2 c1(C(=O)OC)csc(C(C(=O)NCCn2ccnc2)N(C2CCC2)C(C)C)c1 N1(C(c2c(C)cnn2C)C(=O)NCC2CCCO2)CCN(C(C)C)CC1C C1(NC(C2C(C)(Br)C2)=O)CN(c2ncnc3cccc(F)c23)C2CCCCC12 CCC1=C(C(=O)NC2(C)CCN(C(C3(C)CC(F)C3)=O)CC2)CCCO1 C1(NC(CC)=O)CCC(C(=O)NCC(F)CNC(=O)CCOC2CC2)C1 C1(C(N2CCC(CNC(=O)CC3CCOC3)(CO)C2)=O)CC2CCC(C1)C2 CC1CN(C(C2CC2NC(c2c(C(F)(F)F)ncn2O)=O)=O)CCC1O CC(C)(C)CC(C(=O)NCC1CCOCC1)N1CC2CC1CS2 CC1(C(=O)NCCCNC(=O)COCC2CC2)CCCNS1(=O)=O CCC(C)(O)CCNC(C1CCN(C(=O)C(C)N2CC(C)C2)C1C)=O N1(C(c2cnn(C(C)C)c2F)=O)CC2(CC2)CC1CNC(=O)C(C)n1cnnn1 c1(C(C(=O)NCCC)N(C)Cc2ccc(F)c(Cl)c2F)cc2c(cn1)OCCO2 c1(CC(=O)NC(C2CCN(C(c3cc(F)c[nH]3)=O)C2)C)cc(Cl)ccc1O C1(CN(c2nnc(C)o2)C)CCN(C(c2ccc(F)cc2)=O)CC1C c1(CNC(c2cc(C)no2)c2nnnn2CCCC2CC2)cc2cccnc2s1 CS(=O)(=O)C1CC(C(N2CCC(NC(c3cnoc3)=O)C(F)C2)=O)C1 c1(CC(N2CCC(N(C(=O)CNC=O)CC)C2)=O)cc(C)nn1C N1(C(CC=C=C)=O)CCC(C(=O)Nc2ccc3nc[nH]c3c2)CC1(C)C C1(N(C(c2cncn2C)C(=O)NCCC#C)CC)CCCCC1C C(C)(CC(C)NC(C1(N=[N+]=[N-])CC1)=O)NC(CN(S(CC)(=O)=O)C)=O C(c1cccnc1C)=CC(=O)NCC1C2CN(C(c3onc(CC)c3C)=O)CC21 C(c1cn(C)cn1)=CC(N1CCC(C(=O)NCCCn2c(C)ncc2)C1)=O c1(C(N2CCC(CC=C)(NC(=O)C(C3CCC3)OC)C2)=O)ccc(C#C)cc1C c1(NC(c2ccc(NC(C3(Cl)CCC3)=O)nc2)=O)cnc(C(F)(F)F)cc1Cl c1(C(=O)NCC(C)(C2CC2)NC(C(CC=C)OC)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(Cc2c(C)occ2)=O)C(C(N2CC(C)(C#N)C2)=O)CC2CC12 C1(NC(c2cc(SC)c(F)cc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)C1C2 c1(C(=O)NC(c2n(CC)ccn2)C)cc(CNC(c2cc(C#N)c[nH]2)=O)ccn1 CC(C(=O)NCC=CBr)(C1CCC1)NC(=O)Cc1ccsc1 c1(CCC)cc(C(N2CCC(CNC(=O)CSCC(C)C)C2)=O)c(C)o1 N1(C(=O)CSc2ccc(Cl)nc2)CCC2(CC1)CCN(C(C1(O)CCC1)=O)C2 c1(C(=O)NCCC2CCC(NC(CCC)=O)C2)cc(Cl)cc([N+](=O)[O-])c1Cl C1(NC(C2(OC)CCN(C(=O)CCC(C)(C)C)C2)=O)CCn2nnnc2C1 c1(CN(C(C(C)N(C(=O)Cc2ccco2)C2CC2)=O)C)ccnn1C N1(C(C(C)CF)=O)CC2COCCC2(NC(=O)Cc2ccc(C#N)cc2)C1 c1(OCC)cccc(OC)c1C(c1nnnn1C1CCC1)c1cn[nH]c1.CN C1(C(N(CC(O)C2CCC2)C)=O)CCCCCCN1C(=O)CCCNC(N)=O N1(C(C(CCOC)N)=O)CCCC(N=[N+]=[N-])CC1 C(CN=c1nc2sccc2c(N2CCNC(=O)CC2)[nH]1)OCC(C)C N1(C(C(CCSC)OC)=O)CC2CN(C(c3n[nH]c(C)n3)=O)CCC12 N1(N2CC(C#C)(C=O)C2)CC2C3C=CC(O3)C2C1.C(=O)C1=NOC(C)C1 N1(CC2CCCC(OC)C2)CC2(CC(NC(c3cc4ccsc4s3)=O)CO2)C1 c1(OC)ccccc1-c1cc(CNC(N2CC(C(=O)OC)C2)=O)no1 c1(C(N2C(C(=O)NCC3C(C(C)C)C3)CSC2)=O)ccc(Br)cc1 c1(NC)ncccc1C(=O)NCC1C(NC(C2CC(NC(C)=O)C2)=O)C1(C)C C1(NC(c2ccncc2F)=O)CCN(CCCN)CC1.C12(CCCO1)C(=O)NC2 c1(C(C)C)ncc(C(N2CC(O)(CCNC(=O)CCC3CCC(=O)N3)C2)=O)o1 c1(OC)cccc(F)c1C(=O)NCC1CC(NC(=O)CCCc2nc(C)no2)C1 N1(C(c2cc(C#N)on2)=O)CCCCC(NC(c2occ3c2CCC3)=O)C1 C(=O)(C(C)CCOCC(CCOCCC=C)OC)OC C1(NC(c2cccs2)=O)CC=C(C(=O)N2CCCCC2C2CCC2)C1 CC1CN(C(C23CC(CN2C2CC2)C3)=O)CC(C)N(C(c2ccc(=O)n(C)n2)=O)C1 CC(C(=O)N(C1CCN(C(C2CCC(=O)O2)=O)CC1)CC1CC1)C(F)F c1(OC)ccc(CCCC(N2CC(NC(=O)C3CC3)CC2(C)C)=O)cc1OC C#CCC(C)C(=O)N1CC2C(CN(C)C(c3ccncc3F)=O)C2C1 c1(C(=O)NC(CNC(C2C(CC)OCC2)=O)C2CC2)cccc(OC2CCC2)n1 Cc1c(Cl)cc(C(=O)N(c2ncc3sccc3n2)C2CNC2)cc1[N+](=O)[O-] Cc1cc2cccc(NCC34CN(C(=O)OC(C)(C)C)CC3CCO4)c2[nH]1 Nc1ncc(C(N2CC3CC2CN3C(c2ccc(CO)cn2)=O)=O)cc1[N+](=O)[O-] C1(CCN(C(CN(C(C)C)C)=O)C)CCCCN1C(=O)C(C)C1CCCC1 c1(C(N2CC(SC)C(NC(c3cccnc3O)=O)C2)=O)cccc(Cl)c1F Cc1cc(CCC(=O)NCC=CCNC(=O)COc2ccc(O)cc2)nn1C CC(CC(=O)NCCC1CN(C(C2(CO)CCOCC2)=O)CCO1)C(F)F c1(C(N2CCC(O)(CCNC(C3CC4(CC4)CO3)=O)C2)=O)cnc2ccsc2c1 N1(C(C(C)=CC2CC2)=O)CCC(NC(=O)Cn2nnnc2C(C)C)C(O)C1 C1(C)(CC)CC(NC(c2nnn(C)n2)=O)CN1C(c1ccc(OC)cn1)=O c1(-n2c(C(CCCC)OC)nc(-c3cnn(CC)c3)n2)ccc(F)c(C)c1 C(CCCCC(=O)NCC=CCC(N1CCC(CN=[N+]=[N-])C1)=O)N(C)C c1(COCC(N2CCCC2)C)nocc1C(=O)NC1COC(C(=O)OC)C1 C(c1ccc(C(F)F)o1)=CC(=O)NCC1CCCN1C(=O)CCc1ccc[nH]1 c1(C2C(C(N(CC(C)CNC(=O)CC3CCOCC3)C)=O)C2)cccnc1Cl c1(C(N2CC3C(NC(c4c(OCC)ccs4)=O)C3C2)=O)cc2ccc(C)cc2[nH]1 Cc1nc2n(n1)CC(C(=O)N(CCCNC(c1c(C)noc1C(C)C)=O)C)CC2 Cc1cc(C#N)ccc1CC(=O)OC(C(C)(C)C)c1ccccc1 N1(C(C(COCC)NC(c2nonc2C)=O)=O)CC2(COC(C)C2)C1 c1(NC)ccc(CCC(N2CCC(NC(=O)CC(=O)NC3CC3)C2)=O)cc1 c1(C(=O)NC2CCN(C(C3(COC)COC3)=O)C2)ccc(Cl)c2c1OCCO2 C(CC(C(=O)NC1CC(NC(=O)CC2CS(=O)(=O)C2)C1)N(C)C)SC.C(C)N C(N=c1[nH]nc2ccc(Br)cn12)c1ccc(N(C(C)=O)C)c(C2CC2)c1 C(=O)(CCCCC#N)NCC(CN(C(C(c1ccc(C(C)(C)C)cc1)C)=O)C)O Cc1ncc(CCC(=O)OCC23CC(F)C2C3)o1 C(=O)(C(F)(F)CCn1ccnn1)NC(C(C)C)CNC(c1ccno1)=O N1(Cc2ccnc(C(C)(C)C)n2)CCC2(CC1)CC2NC(C1CCN(C)C1)=O Cn1cc(Cn2cc(C(CC3CC3)O)nn2)c(=O)n(C)c1=O C12(NC(c3cncc(SCC)n3)=O)CCCC1CN(C(c1sc(C)nc1C)=O)C2 Cc1cc(CNC(c2cc(CNC(c3sccc3F)=O)ccn2)=O)cc(C)n1 N1(C(CC2(OC)CC2)=O)CCC2(CC1)CC2CNC(=O)C(O)Cc1cnc[nH]1 N1(C(c2c(C)nc(CO)o2)=O)CCCC(C2(NC(=O)C3=CCC3)CC2)C1 C1(CC(=O)NCCC(=C)CNC(c2c[nH]nc2C2CCC2)=O)CCC(C)(C)C1 CC1CN(CCC(C)(C)C)CCC1N=c1[nH]c(N(C)C)nc(=N)[nH]1 C(C)(C)(C(O)CO)C(=O)NCC1(C(=O)NCCc2n(C)ncc2)CC1 C(=O)(CC1OCCc2ccsc21)N1C(COC)(CNC(=O)C2=CCC2)CCC1 N1(C(C(c2cn(-c3nccs3)nn2)CCC)=O)CCOCC(CO)C1 N1(C(C)=O)CCC(C)(C(=O)N(C2CCN(C(=O)CC3(C#N)CCC3)CC2)CCO)C1 c1(C(=O)NC2CN(C(c3c(OC)scc3)=O)C(C)C2)ccc(F)c2cnccc12 c1(C(N2CCC(CNC(c3c(SC)csc3)=O)C2)=O)ccc([N+](=O)[O-])cc1N C=C=C(C)CC(=O)N(C1CCN(C(=O)CN(C2CCS(=O)(=O)C2)C)CC1)C C(CNC(=O)CCCSC)(CCC(F)(F)F)NC(CC1N(CC)CCOC1)=O C(C)(C(C)(C)CC)NC(C1(C)CN(C(C(C)OCCC=C)=O)C1)=O N1(C(CCSCCC)=O)CCC(O)(CNC(=O)C(c2cnn(C)c2)O)C1 O=C1CN(CCCN(C2CCCCC2)C(=O)C(=O)NC2CNCCO2)CCN1 c1(CNC2(CC(=O)NCCCc3ccoc3)CCC2)cc(I)ccc1O C(=O)(C(F)(F)C(C)(C)O)NC(COC)C(=O)NCc1ccc(C)c(C#N)c1 CC(C)CC(C)(C)C(=O)N1CCOC(CN(C(=O)C=CCF)C)C1 C12(C(N(CCC(=O)N(C)CC3CCC(=O)N3)C)=O)CCC(C1)C2 O=C(CCCCC1CC1)NC1CC(CNC(=O)C(C2(O)CCCCC2)(F)F)C1 c1(C(c2nnnn2C(c2ccccc2)C)NCC(C)OCC=C)cc(Br)c(Cl)s1 C(=O)(C(C)(F)C(=O)N(CCC(=O)NCCOCC(C)(C)C)C)OC N(C)(C(=NCC1CCCCC1)NCc1nc(-c2occc2C)n[nH]1)CCC=C C12(NC(C(C=C)N(C)C)=O)CC(CO1)N(C(=O)C(C)CNC(=O)OC(C)(C)C)C2 c1(C(N2CC(C(N(CC(=C)C)CC(=C)C)=O)OCC2)=O)ccc(C)nc1C CC(C(=O)N1CCN(CCCNC(c2cc(F)cc(F)c2)=O)CC1)C(C)(F)F Cc1ccccc1C(C)C(=O)N(CC(O)CN(C)C(c1c(C)ncn1C)=O)C N1(C(CCc2cc(C)no2)=O)CCC(NC(=O)CCC#N)C(C(C)C)C1 N1(C(c2cccc(Oc3cccc(Br)c3)c2)=O)CCOCC1c1ncn[nH]1 C1(CNC(C2(N(C(c3ncn(CC)n3)=O)C3CC3)CCC2)=O)CCOCC1C C1(C(=O)OC(C#C)CC2CCC2)CN(C(=O)OC(C)(C)C)CC12CC2 c1(CC)nnc(C)cc1C(N1CCN(C(=O)C#CC(C)C)C(CO)C1)=O C(=O)(C#CCNC(=O)COc1ccsn1)N(C)CCN1CCCC1 c1(C(=O)NC2CC(NC(C(C)OCCC=C)=O)C2)coc2ccc(C)cc12 CCCC(CCCNC(=O)CCNC(C)=O)NC(c1ccc(F)c(N)c1)=O C=CC(F)(F)C(=O)NCC1CCCN1C(=O)CNC(=O)CN(C)C CCCC(N=c1cc(NCC2CCC3(CCC3)C2O)nc(C(C)C)[nH]1)C1CC1 C1(NC(=O)Cc2c(F)cccc2F)CC2(CCN(C(C3C4CCCC34)=O)CC2)C1 Cc1cc(Br)cnc1C(N1CCN(C(C2CC3(C2)CC(C(=O)NC)C3)=O)CC1)=O c1(OC)cc(CN2CC3CN(C(C4(C#N)CC4)=O)CC3C2)cc(Br)c1O C(=O)(C(C)(CNC(C1CC(C2CCCC2)C1)=O)C(C)C)NCCC(=O)OC CCCCC(CC)CCC(=O)NC(CNC(=O)CCCOCC)C1CCC1 c1(C(N2CCC(NC(c3cc(CC)[nH]n3)=O)C2)=O)cncc([N+](=O)[O-])c1 c1(C(N2CCC(OC(c3cc(C(=O)NC)oc3C)=O)C2)=O)ccc(Br)nc1N c1(C(N2CCCC(N(C)Cc3nnc(S)n3C)C2)=O)cc(S(N)(=O)=O)co1 C(C(=O)N1CC(NC(C2CC3(CC3)C2)=O)C1)(C(C)C)NC(=O)OCC C1(C(N2CCC(NC(C3(C4CCC4)CCC3)=O)C2)=O)CCCC12CCOCC2 CC1CN(C(C2CCN(C(=O)Cc3ccsc3)CC2)=O)CC(=O)N1 C(=O)(N1OC2C=CC1CC2)C1CC(C)N1C(c1cnc(O)c(F)c1)=O C1(CNC(CCCOC(C)C)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC1C1CC1 CCCC(CC)C(=O)N1CCC(C=CC(=O)NC(C)CC(N)=O)CC1 c1(OC)cccc2c(C(=O)NCCOCCNC(C3C=CCS3)=O)coc12 C=CCC(C(=O)N1CC(CNC(C2CNC(=O)O2)=O)C1)OC N1(C(c2c(NC)nccc2)=O)CCC(C)(C(=O)NC(C)COC(F)(F)F)CC1 CN1CC(=O)N(CCCC(=O)N2CC(NC(=O)C(c3ccccn3)O)C2)C1=O Cc1ccc(C(=O)NC(CNC(c2ccc(C(O)CF)cc2)=O)CC(C)C)cc1 C1(CCNC(c2ccn(CC)c2C)=O)CN(C(C2CC(F)(CF)C2)=O)CC(C)O1 C12(C(c3nnnn3C3CCOCC3)NCC(C)OC(F)F)CCC(CC1)OC2.C(CF)O N1(C(C2C(CC)C2)=O)CCCCC2(CCN(C(C34CC5CC3(CO)CC5C4)=O)C2)C1 C1(NC(c2nc(C(C)C)oc2)=O)CN(C(c2n[nH]cc2Br)=O)Cc2nccn2C1 c1(C(C(=O)NCC(=C)C)N(C)CCC2CCCCO2)sc(Cl)cc1Br N1(C(COCCCCC)=O)CCC(C)(CNC(c2c(C(C)C)n[nH]c2C)=O)CC1 N1(C(CC(=C)Br)=O)CC2C(CNC(C3(C)CS(=O)(=O)C3)=O)C2C1 C1(COC)(NC(=O)C=C2CCCCC2)CCN(C(C2(C3CCCO3)CC2)=O)CC1 N1(C(C(CCN(C)C)N(C)C)=O)CC2CCN(C(c3ccsc3Cl)=O)CC2C1 c1(CC)ccc(C(N2CC(NC(=O)C=C(C)C)CC2(C)C)=O)cc1F CC(Cn1ccnc1)C(=O)NCC(CO)NC(=O)C=C1CCC1 C1(NC(C2(O)CC2)=O)CC2CCC1CN2C(c1cc(OC)no1)=O.CCOC N1(C(C(C)N=[N+]=[N-])=O)CCC2C(CCCN2C(c2cccc(N(C)C)c2)=O)C1 CCC(CCOC)C(=O)NCC1(F)CCN(C(C2(C)COC(=O)N2)=O)C1 c1(N2CCC(=CC(=O)NC3CCCCC3)CC2)cccc([N+](=O)[O-])c1 C(C(C(=O)NOC1CC1)C(C)(C)C)NC(C(CC)SC)=O C1(CNC(C(CO)N(C)C)=O)CC2CCC1N(C(=O)C=Cc1cccc(O)c1)C2 c1(N2CCOCC(NC(C(C)SC)=O)C2)ccn2c(Br)cnc2n1 C(=O)(C(C)(C)C1=CCN(C(C2CCCSC2C)=O)C1)N1CC(O)(CCC)C1 Cc1cc(C(N2CC(CNC(=O)Cn3c(C)ccc3C)C(C)C2)=O)c(Cl)cc1F CC(CCC=C(Cl)Cl)N(CCNCCCOC)C C(CN=c1[nH]c(C)nc(=N)[nH]1)(C1(NC(C2CCSC(C)C2)=O)CCCCC1)OC c1(OC)nccc(=NC(c2ccccc2F)c2nnnn2CCC2CC2)[nH]1 Cc1cc(C)c(CC(N2CC(C3CN(C(c4cnccn4)=O)C3)C2)=O)c(C)c1 c1(C(=O)NCC2(F)CC(NC(C(CCC)OCC)=O)C2)c(F)cncc1Cl C=CCC(C)(CC)C(=O)NC1CC(CC(=O)NC2CC3C=CCC(C2)C3)C1 CC1(C)CC(NC(=O)C(=O)NCCC(N)=O)CN1C(=O)C(C)(O)C1CC1 Cc1c(Br)ccnc1C(N1CCN(C)CC1CNC(=O)COCC(F)F)=O C1(C(N2CC(NC(=O)CCCCN3CCOCC3)C2)=O)CC12CCCCCC2 N1(C(C2(OC)CCSCC2)=O)CCC(C2(NC(c3csnc3C)=O)CC2)C1 N1(C(C(CC(F)F)NC(C2ON=C(C)C2)=O)=O)CC(O)C2(CCCC2)C1 C1(C)(C(N2CCC(N(CCC)C(c3ccoc3Cl)=O)CC2)=O)CCC(C)(C)CC1 c1(C(=O)NCCC2C(C(=O)OCC)C2)cc(C2CC2)cc(Cl)n1.c12ccnn1NC2 Cc1nc(C(=O)NC2CN(C(c3ncccc3O)=O)CC2F)ccc1F c1(C(=O)NCC(CC)NC(c2cnn(-c3ccccc3)c2)=O)ccc(C2CC2)o1 CC(C)C(CCN(C)C(=O)Nc1cc(C2CCOCC2)no1)N(C)C c1(OC)ncc(Cl)c(=NC2CCCC23CN(c2nc(C(F)F)nc(=N)[nH]2)C3)[nH]1 C1(CC(=O)NCc2c(C)c[nH]n2)COCCN1C(=O)CN1CCCC1C N1(C(Cc2ccc(C)cc2)=O)CCN(C(c2ccnnc2)=O)C2COCC12 Cc1cc(Cl)c(C(=O)NCC(C(C)C)NC(C2CC(O)C2)=O)cc1F N1(C(CN(C(C2C(CC)N(C)CC2)=O)C2CC2)=O)CCC(C2(C)CC2)C1 C#CC1(C(N2CCN(C(C3CC(OC(F)F)C3)=O)CC2)=O)CCOCC1 c1(C(N(CCNC(C2CCCN(C(C)=O)C2)=O)C2CC2)=O)cnc2c(c1)CCC2 N1(Cc2c(-c3cccc(OC(C)C)c3)cccc2)CC(C)CC(C)C1 C1(CNC(c2cc(I)on2)=O)CCCN1C(=O)C(F)C1CCC1 Cn1c(O)nc2cc(C(N3CCC(CNC(=O)COCCCF)CC3)=O)cnc12 N1(C(CC(CC)CC)=O)CCN(C(=O)CNC(=O)CN(C)C)CC(O)C1 N1(C(CC(CCSC)O)=O)CC2CC3CC2C1C3NC(c1cocn1)=O N1(C(C(C(CC)O)C)=O)CC2CCC1CN2C(c1sc(F)cc1C)=O CC1CC(CNC(c2ccc(C(F)(F)F)nc2)=O)CN1C(c1ccc(O)cn1)=O N1(C(CC2(C)CCN2C(=O)C=Cc2cocn2)=O)CC2C(C1)C2(F)F C1(NC(c2nc(C(=O)OC)oc2)=O)CN(C(C2C3CCCC23)=O)CCC1C C1(N(C(CSCCN(C)C)=O)C)CCCN(C(=O)Cn2cc(Br)cn2)CC1 C1(Cc2onc(C3(COC)CCCC3)n2)CC(N)CC(C)(C)C1 C(=O)(CC(C)(C)C#N)N1CCCC(N(C(C(C)Cc2cnn(C)c2)=O)CCO)C1 CN(C)N=Nc1ccccc1C(=O)NCC1(C(F)F)CCN(C(=O)CO)C1 c1(N2CC(CC=C)(NC(=O)C(C)SC(F)(F)F)C2)cc2nncn2cn1 C(=O)(C(O)CC(F)F)N(C)CCc1cn(CCSc2cccc(Cl)c2)nn1 C1(COC)(NC(C2COCC(C)(C)O2)=O)CCCN(C(c2ccco2)=O)C1 c1(CCNC(C(C)N(CCC)C(c2c[nH]cc2CC)=O)=O)cnn(C)c1C N1(C(C2N(C(c3c(OC)cccc3Br)=O)CC(C)C2)=O)CCCC2(CCOC2)C1 C1(C(N2CCC(C(C)C)C2)=O)CCCCN(C(=O)Cn2cncn2)C1 c1(NC(C2C(NC(c3ccc(C)cc3Br)=O)C2)=O)ccc(Br)c(F)c1CO N1(C(c2c(OC)scc2)=O)CC2(CCCCC2)CC1CO C(=O)(CS(=O)c1ccc(Cl)cc1)N1C(C2CCN(C(C3C(C)C3)=O)C2)CCC1 Cc1cccc(OCCC(=O)NC(C2CCOC2)CNC(=O)CCC=CBr)c1 c1(C(=O)NC2COCCN(C(C3C(C)C3)=O)C2)nn(C)c2ccccc12 C1(CNC(CC(CC)C)=O)CC12CCN(C(c1coc(C(F)F)n1)=O)CC2 N1(C(c2ccc(CC(CC)N)cc2)=O)CCC(O)(C2(C(=O)OCC)CCC2)C1 C1(NC(COC)=O)CCCC1(C)NC(=O)CCOC(C)=O.C(C(F)F)O c1(OC)ccc(-c2nc(CP(C)(C)=O)n(CC3COC(C)(C)C3)n2)nc1 C1(C(N(C2CNC(=O)C2)C)=O)N(C(c2cccc(F)c2)=O)CCC1(C)C Cc1ccc2nc(N3CCCC(C(=O)O)C3C)[nH]c2c1 C1(NC(c2cc(C#N)on2)=O)CC2CC1N(C(=O)CSc1cccc(Cl)c1)C2 C1(CC)CN(C(c2nc(O)sc2C)=O)CCC1NC(c1nnn(C)c1C)=O C1(NC(c2cnc(C(C)C)s2)=O)CC(CNC(c2ccc(O)nc2)=O)C1(C)C CP(C)(=O)CCCNC(C1CC(F)CN1C(=O)C=CCN1CCC1)=O CC1CN(C(c2cnc(Cl)n2C)=O)CC1NC(c1ccc(C2CC2)s1)=O Cn1cncc1C(O)C(=O)NC1CCN(C(=O)CCc2nc(O)n[nH]2)C1 c1(OC)ccc(C(=O)NC2CC(CNC3(C4CC(C)=NO4)CC3)C2)cc1Br N#Cc1ccnc(NCC2(CNc3cnn(CC4CCCO4)c3)CC23CCC3)n1 C12(NC(CCCC=C)=O)CCCCC1CN(C(c1nccc(OC)c1F)=O)C2 N12CC(C(O)C1)NC(=O)CCC=CC2=O.c1(SC(C)(C)C)scnc1-c1cccs1 C1(C(N(CCCCC=C)C)=O)CCCCC1NC(=O)Cc1sccc1C c1(OC)cccc(CCC(=O)NCC(O)CCNC(c2sncc2C)=O)n1 c1(CC(=O)N(C(C)CNC(=O)C(C)Cc2ccco2)CC)ccn(C)n1 N1(C(c2cc(C)nnc2C)=O)CCN(C)CC(C)C1 C1(Cn2cc(CN(C)CCO)nn2)CC2CCCCC2N1C(c1ccoc1Br)=O C12(C(=O)NC3CCC(CNC(c4c(C)cncc4)=O)C3)CCCC1CC(=O)C2 c1(CC)ncc(C(=O)NCC2(O)CCN(C(C3CCN(C)C(=O)C3)=O)C2)c(O)n1 c1(N2CCC(C)C(CO)C2)nc(=NCCc2ccn(C)n2)[nH]c2ccsc12 C1(CNC(COCCNC(c2c(NC)scn2)=O)=O)CC(C)(C)CCO1 C#Cc1ccccc1CC(=O)NC(C)CCNC(C1CC(C)(CC)C1)=O C(CCCC(=O)NCC1CC2CC2N1C(C1CC1c1ccccc1Cl)=O)SC C1(C(=O)NC(C)CNC(c2ccc(C(F)(F)F)cc2)=O)CC2OC1C1CC21 N1(C(N2CCC2c2ccccc2)=O)CCOC(C(F)(F)F)C1 c1(NC(C(CC2CCCC2)NC(c2ccn(CC)n2)=O)=O)cc(C)c(C)c(C)c1 Cc1ccc(C(=O)NC2(CO)CN(C(=O)C(C(C)C)NCCBr)C2)nc1 CC1CC(C(N2CCCC2CN=c2[nH]nc(C3CCCC3)s2)=O)CCN1C c1(C(N2C3C(CNC(C4C(=C)C4)=O)C(C3)C2)=O)cc(Br)cc2nc[nH]c12 c1(C(=O)NC(CC)CNC(=O)Cc2cn(C)nn2)c(C)nsc1NC CC(C)(C)CC(C(=O)N1CCCC1CNC(N)=O)NC(C1C2CC3C(C2)C13)=O CCC(=O)CCC(=O)NCCOCC(=O)N(C(C)CC(=O)OCC)C c1(C(C2CCCCC2)C(=O)N(CCC(=O)O)CC)ccc(F)cc1.n1(C)cnnc1 N1(CC)CCN(CCO)CC1.N12CCCC1C(=O)NCC2=O c1(OC)cccc(Cl)c1CC(N1CCCC(CNC(=O)CC(C)(C)O)C1)=O C1(NC(c2scc(OC)c2)=O)CN(C(=O)CNC(c2ccnn2C)=O)CC1C N1(C(C2N(C)CCC2)=O)CCCC1(C)C(N1CCC1CC(C)(C)C)=O C1(C(=O)NCCCCN(C(C2N(CC)CCOC2)=O)C)CNC(=O)CC1(C)C C(C)(C(CC(=O)Nc1ccc(F)c(F)c1)NC(=O)C(C)N(C)C)OC C(CCCCO)N(C)C(C1(CNC(=O)CC2C=CCC2)CCCO1)=O C1(C)(CNC(C2CCN(C(C)=O)C2)=O)CCCN(C(c2nc(C3CC3)no2)C)C1 CC(C)CC(C)C(=O)NC(Cc1ccco1)C(=O)Nc1ccc(O)cc1 CC(C)CCCC(C)C(=O)NCC1(NC(c2cc3c(Br)c(F)ccc3[nH]2)=O)CC1 c1(C(N(CCN(C(C2CC(C#N)(OC)C2)=O)C)C)=O)cc2c[nH]cnc-2n1 Cc1cc(C(=O)NC2CCC(N(C)C(c3cscc3C)=O)C2)c(C)s1 c1(C(CNC(C2CC2Cl)=O)NC(c2c(CCC)occ2)=O)ccc(OC)cc1 N1(C(C(CN(C)C)O)=O)CC(NC(C2CC3CCC2C3)=O)C(O)C1 N1(S(C)(=O)=O)CCC(CN2CCC(NC(=O)Cc3n[nH]cc3Br)C2)C1 c1(C(N2CCC(C)(C(=O)NCC3(C)CCCC3)C2)=O)n[nH]cc1[N+](=O)[O-] C1(CC)CN(C(=O)C(=O)Nc2oncc2C)CCN1C(=O)CCn1cc(Cl)cn1 c1(C(N2CCCCC(N(C(c3c(C)nco3)=O)C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(CNC(Cc2c(C)nsc2)=O)COCCN1C(c1csc(-c2ccoc2)n1)=O c1(CC)cnc(C(=O)NCCN(C(c2csc(C)c2C)=O)C2CC2)nc1 N1(C(C(C)(CO)OC)=O)CC2CCN(C(c3cc4ncccc4s3)=O)CC2C1 c1(OCC)cccc(CC(=O)NC)n1.C12CCC(CC1)OC1CCN(C1)C2=O.OC N1(C(C(CC#C)O)=O)CCN(C(=O)C(c2ccc(F)cc2)(C)C)CCC1C C(=O)(C1=CC(O)C(NC(c2ccsn2)=O)C1)N1CCN(C(N)=O)CC1 N1(C(C2(CC=C)CC2)=O)CCC(C)(C(N2CCCC(C(=O)N(C)C)C2)=O)C1 c1(C(N2CCC2)=O)ccc(=NCC2CCC(NC(=O)CC3CC(F)(F)C3)C2)[nH]c1 c1(OC)cc(=O)n(C)cc1C(=O)N(CCO)CCOC1CCN2CCOC1C2 CC1CCc2[nH]nc(C(=O)NCC3CN(C(=O)C4=CCCO4)CC(C)(C)O3)c2C1 Cc1cc(NC(c2ccc(F)c(-c3ccc(N(C)C)c(F)c3)n2)=O)nc(C)c1 Cn1nnc2cc(C(N3CCCOC(C4CC4)C3)C(=O)NC3CCCC3)ccc12 O=S(=O)(c1ccc(N2CC3CCC(C2)O3)cc1Br)NC1CC2CCCCN2C1 c1(C(=O)NC2(CF)CCN(CC(C3CC3)OCC)C2)ccc2c(c1)nnn2C c1(CCC(=O)NC(C)C(C)NC(c2cc(CC(C)C)[nH]n2)=O)nnc(S)nc1O c1(CC)nc(Cl)c(F)c(=NCC2CCCN(C(c3cc4ccccn4c3)=O)C2)[nH]1 N1(C(C(CCC)N(C)C)=O)CCC(NC(c2ccc(F)c(C(C)C)c2)=O)CC1C C1(NC(=O)CCn2cccn2)C2CCC1N(C(C1CC(=O)N1)=O)C2 CCC(C)C(C)C(=O)NC12CC1CN(C(c1ccc(N(C)C)cc1)=O)C2 C12(NC(C)=O)CCCC1CN(C(=O)Cc1cc(C3CC3)no1)C2.c1ccccn1 c1(C(N(CCCCCNC(CCOCC)=O)C)=O)ccc2c(c1)SCC(=O)N2 N1(C(c2[nH]cc(C)c2C)=O)CCC(N(C)C(C2CCC(F)(F)C2)=O)C(C)C1 C1(NC(C(C)OC)=O)CN(CC(O)C(C)c2ccccc2)CC1(C)C CCC(C)(C)C(=O)C(=O)N1CCC(C)(C(=O)NC(C)C(=O)OC(C)C)C1 c1(CN2CC(F)CC(NC(C3(C(=O)OC)CC3)=O)C2)ccc(Br)c(Cl)c1Cl C(=O)(C1CCCc2cnc(C)n21)NC(CC=C)CNC(C1C(C)(C)OC1(C)C)=O N1(C(Cn2cc(COc3cccc(C)c3)nn2)=O)CC2CC(OCC(F)F)C2C1 C=C(C)C(CC(=O)NCCCC(N1CCN(CC)CC1)=O)OCC c1(C(N2CC3CC(NC(C4C(C)(C)CCC4)=O)C3C2)=O)cc2cccc(O)c2[nH]1 c1(C(N2CCN(C(CC3C(OC)CC3)=O)C(C3CC3)C2)=O)cccc2sccc12 C#CCCCC(=O)N(CC(=O)NCc1ncnn1C)C(C)C c1(NC(CCC)C)ccc(S(=O)(=O)NCCn2cnnc2C)cc1Cl C1(C(=O)NC2(C(C)O)CC2)(NC(CCN(CC)CC)=O)CCC(C)(C)C1 C(C(C)CC(C)C)N(C(C)=O)CC1(C(=O)NC2CC(n3ccnc3)C2)CC1 N1(C(C(c2cncnc2)C)=O)CCCC(CNC(=O)CCOCC2CCC2)C1 c1(OC)c(F)ccc(CN2CC(F)(F)CC2C(=O)Nc2cnc[nH]2)c1F C1(NC(C(C)C(C)(F)F)=O)CN(CC(=O)NCCNC(N)=O)c2ccccc2O1 CCCCC(C)(F)C(=O)NC(C)(C)CCC1CCN(C(C2CC=CC2)=O)CC1 C1(CNC(C=CCNC(c2ccc(CC)[nH]2)=O)=O)CCCC(OC)C1 C1(C(=O)OCC)C2CC3CN(C(=O)C(N4C(C)C5CCCCC5C4C)C)C1C3C2 c1(C(=O)NC2CN(C(CCOCC)=O)CC3(C2)CC3)c(C)c(C)c(C)c(C)c1C c1(C(=O)NC2C(N(C)C(C3C=CCCC3)=O)CCCC2)ccc([N+](=O)[O-])cc1Cl N1(C(C2(OC)CCSC2)=O)C2CCC1C(CNC(=O)CC1(C)CCCO1)C2 C1(NC(Cc2c(C)nc[nH]2)=O)CCC(NC(c2coc(C3CCC3)n2)=O)CC1 c1(CCC(=O)NCC2CCCN2C(=O)CC2(O)CCCC2)ccc(Br)cc1F C1(=O)CCCCCCNC(=O)CC2CCCC1CC2N(C1CC=CC1)C CCS(=O)(=O)CC(=O)NCC1CCCC(NC(c2ccc(C(N)=O)[nH]2)=O)C1 C1(NC(c2cncc(C)n2)=O)CC2CCC1(NC(=O)Cn1ncnn1)C2 CC1(C)CC(CNC(C2CCCO2)=O)CN(C(c2cnn(C(C)(C)C)c2)=O)C1 n1(COCC)nc(C)c(CC(=O)NCC(C)(C)Cc2ccccc2)c1C N1(C(C(C)n2cccn2)=O)CC(NC(c2ccc(C3CC3)cn2)=O)CC(C)(C)C1 c1(C(=O)NC(C2CCCN(C(CCC(=C)C)=O)C2)C)cc2c(C)n[nH]c2cn1 c1(OC)ccc2c(C(=O)NC3CCCC3NC(C3CC34CCC4)=O)ccnc2c1 CC(C)C(C)(CNC(c1cccc(C2(C)CC2)c1)=O)NC(C1CC2(CC2)CO1)=O c1(CCC)ccc(C(=O)NC23CC(NC(=O)C(C)SC)(C2)C3)cc1[N+](=O)[O-] C(=O)(CCC(=O)NC(Cc1ccoc1)C(=O)NCCC1COCCO1)NC N1(C(CC=CC=C)=O)CCCC1C1CCCN1C(c1ncc(C)cc1F)=O N1(C(CCc2ccc(OC)cn2)=O)CCC(NC(=O)C(C)SC)C(C)C1 C1(NC(C(C)CO)=O)CCN(C(=O)C=Cc2ccoc2)C1c1ccccc1 C1(N2CCN(CCNC(CCC)=O)CC2)(CO)CCCCC1.C(C)(C)C C1(F)(CNC(=O)CCc2ccc(Cl)s2)CCC(NC(=O)CN2CCCOC2=O)C1 C1(C(=O)NCC(C)CC(=O)NC2CN(CC3CC3)CC2C)C2CCCCCC12 N1(C(CC2C(CNC(c3ccc(C#C)o3)=O)C2)=O)CC(F)(F)CC1CCO c1(OC(CC(C(C)(C)C)NC(C)(C)C)=O)ccc2c(c1)COCC2 c1(CCC(=O)NC(CN(C(CCOC)=O)C)C)c[nH]c(C)c1C(=O)OC C1(C(N2CC(C#C)C(OC)C2)=O)CC2CCCC2N1C(c1cncnc1)=O C1(CNC(Cc2cc(C)on2)=O)CCCC2(CN(c3ncnc(Cl)c3C#N)C2)O1 c1(C(N2C(CNC(c3c(CC)ocn3)=O)CC(OC)C2)=O)cc(C)cc(F)c1 CC1(C)CCC2(CC1)CC2C(=O)NCC1C2CN(C(c3ccsn3)=O)CC12 c1(C(=O)NCC2CN(C(=O)CC3CCCCO3)C2)cc2nc[nH]c2cc1[N+](=O)[O-] C(=O)(CC(C)N1CCCC1)NCC(C)N(C)C(C1C2CCCC12)=O CCC(C)CCCC(=O)NCCOCCNC(=O)CCCCCNC(N)=O N1(C(C(=O)C2CC2)=O)CC2CCC(C1)N2Cc1ccc(F)c(C(=O)O)c1 c1(-c2nc(CCCCCC)nn2CCC)ccc(S(C)(=O)=O)c(SC)c1 c1(C(=O)NC(C(C)O)CO)cn2c(n1)CN(Cc1ccc(C3CC3)cn1)CC2 N1(C(C)=O)CCC(C2CCN(C(c3ccccn3)=O)C2)C1 c1(C(=O)NC23CC(NC(C4C(C)(C)C4(C)C)=O)(C2)C3)ccc2ncccc2n1 C1(NC(C2(C=C)CCC2)=O)CN(C(=O)CN2CCC2C)CC(C)(C)C1 c1(OC)cncc(C(N2CCC(F)(C(=O)N(C3CC3)Cc3cccnc3)C2)=O)c1 C1(N(C(C(CC)OCC)=O)C)CCCCN(C(=O)Cc2cc[nH]c(=N)c2)C1 C1(CNC(=O)CN2CC3CC3C2)C2CN(C(C3(N(C)C)CCCOC3)=O)CC12 C(=O)(C(CC)NC(=O)COc1ccccc1)N1C(CNC(C=CCC)=O)CC1 Cc1cnn(C2CC(C(=O)NCC3CN(Cc4cccnc4)C3)C2)c1 c1(C(N2C(C3(NC(C(C)=C(CC)C)=O)CC3)CCC2)=O)c(Cl)ccc(C)c1O N1(C(c2ccsn2)=O)CC2CCC(C1)N2C(C1CCC2CC1CO2)=O c1(NC(=O)CC2COCC2(C)C)cnn2ccccc12.C1(N(C)C=O)CC(O)C1 c1(CCC(=O)NCC(C)N(C(=O)CCC2CCCN2C)C)cccc(Br)c1 n1(C(C(c2nnnn2C2COC2)NCC(C)C)C)cc(-c2ccccc2)nn1 c1(C(N2CCCC(F)(CNC(C3(C)CC3(F)F)=O)C2)=O)c(Cl)ccc2c[nH]nc12 N1(CCNC(c2cn(C)nc2)=O)CCCN(C(C2CC3(CCC3O)C2)=O)CC1 C1(C(N(CC(C)NC(C(C)N(CC(F)(F)F)C)=O)C2CC2)=O)CC(S(C)(=O)=O)C1 C12(C(N3CC(CNC(C4(OCC)CCOCC4)=O)C(C)C3)=O)CCCC1C2(F)F CCC(C#N)(CC)C(=O)NCC1CN(C(C2CCN(C)CC2)=O)C(C)(C)C1 C1(NC(=O)NC2C(CC)CCCC2)(Cc2ccc(NCC)o2)CCC(F)(F)CC1 C(=O)(C(CCC(C)C)NC(=O)CCCCN(C)C1CC1)NCc1cnc(CC)[nH]1 C1(C(=O)NC(C#CC)(C)C)CC=CCN1C(=O)CC(C)N(C)C N1(C(=O)NC)CCC(Oc2ccc(C(=O)NCC)cc2)CC1.C1(CN)CC1 N1(Cc2cc(Cl)cc(C)c2O)CC(C2CCCN(C(c3cc(Br)c(C)s3)=O)C2)C1 N1(C(=O)C=CCO)CCC2CN(C(=O)COC3CC3(F)F)CC2CC1 Cc1cc(C(=O)Nc2cccc(NC(c3ccnn3C(C)(C)C)=O)c2)nc(O)n1 N1(C(C(CCCC)O)=O)CCC2(CCC(N(C)C(C3CCS3(=O)=O)=O)CC2)C1 c1(OCC)cccnc1C(N1CCCC1CN(C(C12CCCC1C2)=O)C1CC1)=O Cc1cc(CC(=O)NC(C(=O)NC2CC(=O)NC2=O)C(C)O)n(C)n1 C(=O)(CS(=O)(=O)C1CC1)N(C1CCC(NC(C23CCC(CC2F)C3)=O)C1)C C(CC(C)C)(C(=O)NCC1CCCCN(C(=O)CSCc2ccccn2)C1)OC C12(NC(c3c(C)nn(CC)c3C)=O)CCOCC1CN(C(=O)CC1(C)CC1)C2 c1(C(N2CCC(F)(CNC(CN3CC(C)(C)C3)=O)C2)=O)cc(F)ccc1O N12CCCC3CN(CCC13)C2=O.c1(CNC(C)=O)cn2cccc(C)c2n1 n1(Cc2cc(C)no2)nnc(C(=O)NC2CC(NC(C3CCC3)=O)C2)c1C C1(C(=O)NCC(COC)NC(=O)CN2CCC(OC)C2)CC1C1CCC1 C12(CNC(c3cc(CC)nn3C)=O)CCC(C1)N(C(=O)C(C)SC)C2 C1(NC(c2c(OC)cnc(Cl)c2)=O)CCN(C(=O)CC23CC(C2)C3)CC12CCC2 Cc1nc(C(=O)NCC(CO)NC(c2c(C)cc(C)cc2C)=O)ccc1C#N C(=O)(C(C(=O)NC(CNC(=O)Cn1nccn1)C1CC1)C(C)C)OCC C1(C(N(CC(CCC=C)O)C)=O)CC(C)CCN1C(=O)C(C)N1CCCC1 N1(C(Cc2nnc(C)o2)=O)CCC(NC(=O)C(c2cccnc2)O)C(C)C1 N1(C(c2ccc(Br)nc2)=O)CC(C(N2CC3CCCC3C2)=O)CC(F)(F)C1 c1(CC(=O)NC(CCOC)CNC(C2CC=CC2)=O)ccc(OC)c(Br)c1 c1(C(=O)NCC(C)C(=O)NC2(C)CCCCC2)n[nH]c2c1CCC2 c1(NC(C2C(NC(C)=O)CCC2)=O)cccc(Cl)c1[N+](=O)[O-] CC(CC(=O)N1CCC(C(C)NC(n2cc[n+](C)c2)=O)C1)C1CC1 C1(CNC(C(C)CC2CC2)=O)CCC(OCC(F)F)CC1.C1(=O)C(C)(C)CN1 CN1CCC(C)(C(=O)NC2C3CC4C2C4C3C(=O)NCC2CCCC23CC3)CC1 CCC(CC)(C(=O)NCC1CCN(C(c2nnn(C)c2C(F)F)=O)C1)C(C)C c1(OC)ccc(C(=O)N(C)Cc2cn(CCSc3cc(C)n(C)c3)nn2)c(Br)c1 c1(C(=O)NC2CC(NCc3cn(C)nc3)C2)cc2nccnc2cc1F C1(C)(C(=O)NC(C)CN(C)C(c2ccco2)=O)CCCCC1(F)F Nc1cc2ccccc2c(C(=O)NC2CC(CNC(C3CC(F)C(=O)N3)=O)C2)n1 N1(C(C2C(C#N)C2)=O)CCCCC1CCC(=O)N(CCCCCN1CCCC1)CC C1(C(N2CC(C)(C)OCC2)=O)N(C(C2CC2[N+](=O)[O-])=O)CCCC1(C)C Cc1ccc(O)cc1C(=O)NC(CO)C(C)NC(=O)Cn1nc(C)c(Cl)c1C Cn1c(=O)cc(C(=O)NCCNC(c2cc(C(=O)O)on2)=O)c2ccccc12 c1(C(=O)Nc2cnc(CCCC)nc2C)cc(S(N)(=O)=O)cn1C N1(C(c2cn(CC)nn2)=O)CCOC(C(C)NC(c2ccc(Br)o2)=O)C1 CC1CCCCC1C(=O)NC1CC(NC(=O)C(C)(F)F)C(O)C1 c1(CC(=O)NCC2CN(C(C3C(C)CC3)=O)C2)csc(C(F)(F)F)c1 C=C=CCC(=O)NCCOCCCNC(=O)CC1(C)CCCO1 N1(C(C=CCN(CC)CC)=O)CCCC(N(C(=O)C=C(Cl)Cl)C)C1 N1(C(CCc2cc(C)on2)=O)CCN(C(c2cccn(C)c2=O)=O)C(C)C1 CC(C)CCCCC(=O)N1CCN(C(=O)CCCSc2ccccc2)CC1C c1(C(=O)NCCC(=C)CNC(C2(OC)CCSC2)=O)cc(C)c(F)cc1F c12cnccc1Cc1ccc(cc1)-c1cn-2nn1.C1(C(N)=O)CN(C(=O)N(C)C)C1 C1(CC)CCC(C(c2nnnn2C2CCC2)NCCCCCOCC)C1 CCCC(C)C(=O)N(CCCN(C(=O)CCc1ccc(SC)cc1)C)C c1(N2CCC(NC(c3cnc(SC)nc3O)=O)C(C)C2)ccc([N+](=O)[O-])cc1F C(C1CCCCc2ccccc21)NC(Cn1cc(-c2cc(C)c(F)nc2)nn1)=O c1(OC)cc(OC(C)(C)C)c(CNC(C23COC(CO)(C2)C3)=O)cc1NC(C)=O CC1CCn2cc(C(=O)N(C3CN(C(c4cnc5nccn5c4)=O)C3)C)nc2C1 C1(NC(C(C)OC)=O)CCCN(C(c2ccc(-c3ccsc3)cc2)=O)C1C c1(CCC(N2CCN(C(=O)COC3CCOC3)CC2)=O)c(F)cccc1F O=C(C1=COCCC1)NCC1CN(C(=O)COCC2CCCO2)CC1(F)F c1cccc(Cl)c1C.C1(C(=O)OC)CC(C(=O)N2C(=O)N2)C1.C(CC(C)O)CCN c1(C2C(NCc3cccc(OC)c3)C2)c(Cl)cccc1Cl N1(C(C(C)NC(N)=O)=O)CCOCC1CN(C(=O)C(F)(F)c1nccs1)C C1(C(N2C(CNC(c3n(CC)ncc3)=O)COCC2)=O)CCOCC12CCC2 C1(C(=O)NCC2(CCN(C(C3CC34CCC4)=O)C3CC3)CC2)COCC1C(N)=O C#CC(C)(C)C(=O)NC(C1CCN(C(c2c(C(F)F)ncn2O)=O)C1)C c1(C(=O)NC(C)CCNC(C2CC(O)C(F)C2)=O)ccc2nc(O)n(C)c2c1 N1(C(CCC=CCC=C)=O)CCN(C(=O)COCc2ccccn2)C(CCO)C1 C1(C(=O)NC2CCC(CNC(CCCNC(=O)OC)=O)C2)CCC(=O)N(C)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(C)CCCN(C(CSSC)=O)C1 N1(C(C(CC)OCC)=O)CCC(NC(=O)C(C)C2CCOC2)C(C)(C)C1 N1(C(CC2OCCN(C(c3c(C)snn3)=O)C2)=O)CC2CCC1C(O)C2O CC(CC(=O)NCC1CCCCN(C(=O)CS(C)(=O)=O)C1)CC(F)(F)F CC(CCCNC(=O)C=CCc1cn(C)nn1)NC(=O)CCC1CCCCO1 c1(CC)cc(C)ccc1C(=O)NCCCC(C)NC(=O)CSCC(=O)OC CCN=c1[nH]cc(C(N2CC(NC(=O)CCNC(C3CC3C)=O)C2)=O)s1 C(CN=C(NCc1cc(C(C)(C)C)on1)NCC1CCC(C)O1)SC Cc1cc(Br)c(CN(CCc2ccccc2)Cc2cnn(C)c2)s1 n1(CC(=O)N(CC(CC)NC(=O)C(=O)C2CC2)CC)nc(C(F)F)cc1C(F)F N1(C(C2(COC)CCC2)=O)CC2C(NC(C3CCCOCC3)=O)CS(=O)(=O)C2C1 c1(C(=O)NCCNC(C2(C(F)(F)F)CC(F)C2)=O)cc2cc(F)c(F)cc2[nH]1 N1(c2ccnc(C)n2)CCC(C2CC2)(CN(C(=O)CC2(C)CCS(=O)(=O)N2)CC)C1 N1(C(C2C(C(=O)OC)C2)=O)CCC(C(F)C(=O)NCC2CC3(CC3)C2)C1 CCC(CC(=O)N1CC(OCCC(=O)NC2CCOCC2C)C1)C1CCC1 C(=O)(CCCC#N)N(CCC(N1CC(C)(F)C1)=O)CCO N1(C(Cc2c(C)ccs2)=O)CCCC(O)(CNC(=O)CCCc2cnccn2)C1 C12(C(F)(F)F)CCCN(C1)C2=O.N1(C(COC)=O)CCC(CC(=O)OC)C1.C(C)(=O)O C#Cc1ccnc(C(=O)N(C2CCN(C(=O)CSCCC(F)(F)F)C2)C)c1 C12(C(=O)NC(c3ncccn3)C)CC(CO1)N(C(=O)Cn1ccnn1)C2 C1(CNC(CC(CCC)O)=O)CCC(C)(C)CN1C(=O)Cc1cc(C2CC2)no1 c1(OC)ccc(C(=O)NC2(n3cc(-c4nccn4C)nn3)CC2)cn1 c1(CC)conc1C(=O)N(C(C)(C(=O)NCC1(C(N)=O)CC1)C1CC1)C C(=O)(CC(C(C)(C)C)NC(C1CCC(C)(C)CC1)=O)NCC1(COC)CCCC1 C1(NC(c2cnccc2Cl)=O)CC(CNC(=O)C(Cl)=CCl)C12CCC2 C1(C(N2C(CC)(CC)CC2)=O)CCN(C(=O)C(c2ccn(C)n2)C)C1C C1(NC(CCCC(N)=O)=O)CCN(C(c2cc(C(N)=O)cc(F)c2)=O)CCC1CO C1(NC(C(C)Cc2ccccc2Cl)=O)CC2(CCN(C(=O)Cn3cccn3)C2)C1 c1(OC)cnc(Cl)cc1C(N1CCCC(C)C1CNC(c1ccnc(O)c1)=O)=O c1(C(=O)NC(CCCCNC(C2C(C)C2)=O)C)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2C(NC(=O)CCOC3COC3)CC2)ccc(F)cc1 Cc1ccc(NCC2CC3CCC2N3C(=O)CCC(C)N(C)C)c([N+](=O)[O-])c1 C=CCN=C(NCC1(O)CC2CCC1C2)N1CCC(O)(C#C)C1 N1(CC(=O)NCC=C)CCOC(c2cn(CC3CCCNC3)nn2)C1 C1(C(N(C)CC2CC(F)CN2C(c2ncccc2Br)=O)=O)CC(=O)NC(=O)C1 Cc1ccccc1CC(C1CCNCC1)NC(=O)Cc1csc(-c2ccoc2)n1 C12(CC(=O)NCCC3CSCCN3C(=O)CN3CCSCC3)CNC(=O)C(C1)C2 N1(C(CCCC)=O)CCN(CCNC(=O)Cc2ccc(F)c(F)c2)C2(CCC2)C1 C1(CNC(COCCC=C)=O)CN(C(c2cc(C)oc2CC)=O)CC1C(F)(F)F CC(C)C(C)C(=O)NCCC1CCN(C(=O)C(Cc2ccsc2)N(C)C)CC1 N1(C(C(c2n(CC)cnc2)=O)=O)C=C(Br)CC(C(=O)OC(C)(C)C)C1 C1(CNC(CC(C)n2cccn2)=O)CN(C(c2cc(Cl)nn2C)=O)CCN1C Cc1cc(C(c2nnnn2CC2CCCO2)NCC2COCCO2)nc(Cl)c1Br C1(CNC(CCCC)=O)CC(NC(=O)CC2CC(=O)NC2=O)C(O)C1 N1(C(CN(C(C)C)C)=O)CC(CNC(=O)C(C)Cc2cnc[nH]2)CC(C)(C)C1 CC(C)CC(C)CC(=O)NCC(CNc1ccc(C(F)F)cn1)CC1CC1 Cc1ccc(C)c(C(=O)NC2CC(F)CN(C(=O)Cn3c(C)c(C)sc3=O)C2)c1 CCCCCCN(C1CC(C)(NC(=O)Nc2nsnc2O)C1)C c1(C(N2CC(C)(NC(C3CCN(CCC)CC3)=O)C2)=O)cc2cccnn2n1 N1(C(C)C)C(=O)CCC1C(=O)NCC1CC(O)CN1C(=O)CSc1n[nH]c(O)n1 C1(NC(C(C(C)C)NC(c2c(CC)[nH]cc2)=O)=O)CC(F)(F)C1(C)C C12CCC(CC1)C(=O)N2C.n1(CCCNC(=O)Cn2cccc2)ccnc1 Cc1cc(F)cnc1C(=O)NC(CC(N)=O)C(=O)N(C)C(c1ncccn1)C C(CC(CNC(=O)CC1(C)CC1)OC)NC(C(C)SCCCC)=O c1(SC)nc(N2CC3CC(NC(=O)C(C)(F)F)C3C2)cc(C)n1 N1(C(Cc2cc(C)no2)=O)CC2CC1(CNC(C1CC1(Cl)Cl)=O)C2 c1(OC)cc(SC)ccc1C(=O)NCC1CCC(CNC(=O)C(C)C(C)C)CC1 C(C(CC(=O)NCc1cccnc1)C1CCC1)NC(c1c(C(C)C)[nH]cc1)=O CC1(C)CCN(C(c2ccc(=O)oc2)=O)CC1NC(C1CCCSC1)=O Cc1cccc(C(F)C(N2CCC(O)(CN(C)C(c3ccc[nH]3)=O)C2)=O)c1 C12(Cc3c(NC(=O)C(=O)NC4CSC4)ncs3)CC3CC(CC(C3)C1)C2 C(c1cccc(F)c1)=C(C(=O)NCCC1(NC(C(CC)O)=O)CC1)F c1(N(C)C)ccc(C(=O)NC2CCCC(N(C(=O)C=Cc3cn[nH]c3)C)C2)cc1 CC(CN(C)C)CC(=O)NCC1CCN(C(C2CN3CCN2CC3)=O)CC1 c1(C(=O)NCC2C(NC(C(C)N3CCC3)=O)COC2)ccc2cc(O)ccc2c1 C1(CNC(C2(COC)CC2)=O)CC2CCC1N(C(=O)CCc1nncs1)C2 c1(C(CCN)=O)ncnc(N2CC3C=CC2C3)c1Br.c1(O)ccc(Cl)nc1 N1(C(c2ccc(N(C)C)cn2)=O)CCN(Cc2ccc(Br)cn2)C2CC12 c1(N(C)C)csc(C(=O)NCC2CCN(C(C3(C(F)F)CCCO3)=O)C2)c1 c1(C(N(CC(CC)NC(c2sc(C)nc2C(C)(C)C)=O)C)=O)ccc(C)cc1 c1(CNC(C2C(C)CC2)=O)cc(C(=O)NCCOCC2CCCC2)n[nH]1 C1(CC(=O)NC)CN(C(=O)CCC(N)=O)CCN1C(c1cc(N)nc(Br)c1)=O C(=O)(CCC(C)N(C)C)N(CC(C)O)CCNC(COCC#C)=O CC(C)(F)CCC(=O)NC1(C(N2CCC(C(F)F)CC2)=O)CC1(C)C Cc1ccn(CC(N2CCC(C(C)(C)NC(c3ccc[n+]([O-])c3)=O)C2)=O)c(=O)c1 C(=O)(C1CCCn2ccnc21)NC(CC)CNC(=O)CC1CC(OC)C1 C(c1cnc(O)nc1O)=CC(=O)NCC1(O)CCCN(C(c2csc(Cl)c2)=O)C1 CC1(C)CC(NC(c2cccc([N+](=O)[O-])c2)=O)CN(C(C2CCC(=O)O2)=O)C1 CC1CCC(C)(NC(C2(C)CCCN2C(=O)CN2CCC(=O)CC2)=O)C1 O=S(=O)(c1ccc(NCC2CCCC2O)c2cnccc12)N1CCOCC1CO Cc1cc(C(C)C)c(C)o1.C12CCC1N(C)C2 N1(CCC)CCCC1C(=O)NCC1(O)CC(C(N2CCC2CN=[N+]=[N-])=O)C1 C1(CC(N2CC(OC(CC)=O)C2)=O)CN(C(C2(C(N)=O)CC2)=O)CC12CC2 C1(NC(=NCC=C)NCc2cn(CC=C)nn2)COC2(CCOCC2)C1O C1(C(N(C2(C(N3CC(C(C)(C)C)C3)=O)CCC2)C2CC2)=O)CCOC(=O)CC1 C1(F)(NC(c2nc(-c3c(C)cccc3)c(C)s2)=O)CCS(=O)(=O)C1 CC1=NS(=O)(=O)NC=C1C(=O)N1CCN(C(=O)CSCC(N)=O)C(C)C1 C1(CNC(CCC)=O)CC(C)N(C(=O)C=Cc2cn[nH]c2)C1 N1(NCC2(CC(F)F)CCCC2)CCN(Cc2cnc(N3CCOCC3)s2)CC1 CCC(C(=O)Nc1nc(CO)cs1)N(C(C)C(=O)OC)C1CC1 N1(C(c2cncc(OCC)c2)=O)CCOCC(NC(c2cc(C(F)F)on2)=O)C1 C12(NC(C3CC(OC)C3)=O)COC(C1)C(NC(=O)C(C)c1ccsc1)C2 C(=O)(CCCCN(C)C)NCC(C)C(=O)NCC1CC1c1ccoc1 N1(CC2CCCC(OC)C2)C(=O)CCN(Cc2ccnc(-n3cncn3)c2)C1=O C12(C(=O)NC3COC3)COC(C(=O)Nc3ccc(Br)cc3)(C1)C2 C1(CCOC)(C(N2CC3C=CC2C3)=O)CCN(c2ncc(Cl)cn2)CC1 C#Cc1cc(C(N2C3CCC2CC(N(C)C(C2CC2C(F)F)=O)C3)=O)cc(F)c1 c1(OCC)ccnc(NC2CN(CC(F)F)C2)n1 N1(C(C2N(C)C(C(N)=O)CC2)=O)CC(CNC(C2CC2C(F)F)=O)OC(C)(C)C1 C(=O)(CCCc1csc(=N)[nH]1)N(CC(C)CNC(C1COCC1C(F)(F)F)=O)C C1(C(C)OC)CCN(C(=O)CN(C2CCCCC2)C(=O)CSC(C)C)C1 C1(O)(CCNC(c2c(C(N)=O)coc2)=O)CCCN(C(=O)C2=CCCCO2)C1 c1(C(C)NC(=O)C(=O)Nc2cnc(C3CC3)nc2)ncccc1F CCCCC(C)C(C(=O)NCCN1CCCCC1)N1CCC(CC2CCC2)C1 C(C)(N=c1nc2c(cnn2C)c(N(C)Cc2ncn(C)n2)[nH]1)c1n(CC)ncc1 c1(OC)cncc(NCC(=O)NCNC(=O)C(N)=O)c1 c1(C(=O)NCCCN(C(C2(C)C(C)OCC2)=O)C)ccc2cc(Br)ccc2c1 c1(C(=O)NC(CC2CCN(C(CCN(C(C)=O)C)=O)CC2)C)ccn2ccsc12 c1(C(=O)NCC(n2cc(C(C3CC3)NC(C3CC3)=O)nn2)C)ncccc1O N1(C(C(CC)n2ccnc2)=O)CCC(C(C)(C)C)(CNC(=O)COCC(C)C)C1 C12(C(=O)NCC(=O)NC)CCCC1CCN2C(C1CCS(=O)CC1)=O C1(CC=C)(NC(=O)C=CC(N)=O)CCCN(C(c2cc(Cl)ncc2F)=O)C1 C1(C(=O)NCC(C)CNC(=O)CCc2cncs2)CC12CCCC2 c1(C(=O)NCCCCNC(c2cc(F)c(CO)c(F)c2)=O)cc2cn[nH]c2cn1 CC1CCC(=CC(=O)NCCC(O)CNC(C2CC2c2ccccc2F)=O)CC1 c1(CC)conc1C(=O)NCCn1ccc(C(=O)N(C)CCN(C)C)c1 C1(C(N(C(C)CO)C)=O)CCCN(Cc2cccc(Br)c2)C1 CC1(OCC(=O)N(CCCO)CCO)CN(C(=O)C=Cc2cocn2)C1 c1(C(=O)NC2C(NC(C3(C)CC=CCC3)=O)CCC2)cnnc2ccccc12 C(=O)(C(C)(C(F)(F)F)NCC(=O)NCCC(C(C)C)C)NCC(=O)OC(C)(C)C C1(C(c2n(CCOC)nnn2)NCCc2ncnn2C)CCCCCC1 c1(C(=O)NC2CN(C(c3cc(C)cc(C)n3)=O)C2)ccc2c(Br)cccc2c1 c1(CC(=O)NCCOCCNC(C(C)SCCCC)=O)ncoc1COC Cc1ccccc1CNC(c1nnnn1C1CC1)c1cnoc1 Cc1ccc(CO)c(-c2nn[nH]n2)c1.C(CC(C)C)(C(=O)N1CC=CCC1C)N N1(C(C(CC=C)C)=O)CCC(C)(C)C(NC(=O)Cn2ccc(C)n2)C1 N(C1COc2ccc(S(C)(=O)=O)cc21)C(N1CCC(C(CC)CC)C1)=O Cc1nc(CC(=O)NCC2OCCC2C(=O)NC2CC2c2ccccn2)n[nH]1 N1(C(C2C(C)(Br)C2)=O)CCC2(CCN(C(=O)C(=Cc3c[nH]cn3)F)C2)C1 C(C(=O)NCCC1CC(C(N2CCCC(C(N)=O)C2)=O)C1)(C(C)C)OCC C(N=c1cc(NCCCCCO)nc(C2CC2)[nH]1)c1c(=N)cc[nH]c1 Cn1ncc2c(C(N3CCN(C(=O)CC4CCC4)CC34CC4)=O)ncnc12 c1(OC)cc(CN2CCCC(CNC(=O)C(n3cc(C)cn3)C)C2)ccn1 Cc1cc(NC(CNC(C2CCC3CC3CC2)=O)C2CCC2)n2nc(C)cc2n1 c1(C(=O)NCC2CN(C(C(C)OCC)=O)CC2O)ccc(Cl)c(O)c1N c1(SC)cccc(C(N2CCCCC2CCNC(c2cncn2C)=O)=O)c1 CC1(CNC(C2CC2c2cccs2)=O)CCN(C(=O)CCN2CCOC2=O)CC1 CC(C)C(CNC(=O)C(C)(C)Cl)NC(C1CC(C(F)(F)F)C1)=O N(C(=NCCC(=O)N(C)C)N1CC(F)(F)C(F)(F)C1)CC1(C)CCC(F)(F)CC1 c1(C(=O)NCC(CC)(CC)NC(=O)Cc2nocc2C)cc2cnccc2o1 Cc1ccn2cc(C(=O)NCC3CC(F)(F)CN3C(c3oncc3C)=O)nc2c1 CC1CN(C(=O)CN2CCOCC(SCc3ccn(C)n3)C2)CC(C(C)C)O1 n1(CC(=O)NC2(C)CC(NC(c3cc(C(C)C)[nH]n3)=O)C2)cc(P(C)(C)=O)cn1 C1(CC)CN(C(c2csc(-c3ncccn3)n2)=O)CC1NC(c1cnoc1C)=O c1(C(C(=O)NC2CC2)N(CC)CC2CCOC2)ccc(-c2nc(=O)o[nH]2)cc1 c1(C(N2CCC2c2cn(Cc3ccnc(Cl)c3)nn2)=O)cccc2ncccc12 CCC(C(=O)N1CCCCC1CCN(C)C(c1cc(Cl)sc1Cl)=O)C(C)C CC(C)CC(C)OCCC(=O)N(CCNC(c1cc(C2CC2)on1)=O)C1CC1 N(C(=NCC1CCSCC1)NC1CCC1)C1CCN(C(N2CCCCC2)=O)C1 C1(=O)C(C2(CNC(=O)CSC)CC2)NCCN1.C1(C(C)CC)(C(=O)NC)CC1 C(=O)(C(CC(F)F)NC(=O)CC=CCCCCC)N(CC#C)C C1(C(=O)NCCSCC)C2CC2CN1C(c1ccccc1C)=O C(N=c1cc[nH]cc1S(=O)(=O)NC1CCN(CC(C)C)C1)c1ccc(SC)nc1 c1(C(C)NC(C2CC2NS(=O)(=O)c2nccs2)=O)ccc(Br)cc1F N#Cc1ccc(C(N2CC3(NC(C4CC4(F)F)=O)CC2C3)=O)cc1 NS(=O)(=O)c1ccc(Cl)c(S(=O)(=O)NC(c2cnc3c(c2)c(O)nc(=O)n3C)=O)c1 CC(CC(=O)c1ccc(F)cc1)C(=O)N1CCC(NC(=O)CCC2CCC2)CC1 N1(C(C(C)N(C)C)=O)CCC2(CCCCC2NC(C2CCC3CC3C2)=O)C1 C1CCC(=O)N1.c1(CC(CSC)NC(=O)CC)ccccc1.N(C)(CC)CC c1(C(c2n(CC(F)(F)F)nnn2)NCC2(CCCO)CC2)cc(Cl)cc(Br)c1F c1(OCC)ccc(CC(=O)NC(C)C(CO)NC(=O)C(C)OC)cc1OC CCCCC(C)C(=O)N1CCCCC(CNC(c2ccoc2C(C)C)=O)C1 Cc1ccccc1OCC(N1CC(NC(C2(C)CCCO2)=O)C(CC2CC2)C1)=O C1(C(=O)NCC2(CCS(N)(=O)=O)CC2)CC2(CCC2)CN1C(=O)CC1=CCCC1 C1(NC(COc2cccc(C)c2)=O)CN(C(C2CSCC(=O)N2)=O)CC2(CC2)C1 N1(CCc2ccc(N(C)C)cc2)C(=O)NC(Cc2ccnn2C)C1=O C(C(CC(C)C)C(=O)NCc1cc(C(C)C)no1)NC(c1c(NC)cccc1)=O N1(C(C2C3CN(C(C4CC(C)C4)=O)CC32)=O)CCC(CO)C(O)C1 C1CCC(C)(C)C(=O)N1.Cc1nccn1CC(N1CCC(N2CCCC2)C1)=O c1(C(N2CCC(COCC)(OCC(=O)OC)C2)=O)n[nH]c2ccc(Br)cc12 Cc1c(NC(=O)CN2CC3CCC2C3)ncnc1N1CCOC(C(N)=O)C1 C#Cc1ccc(C(=O)NCC2CCCCN2C(=O)C(C2CCOCC2)C)cc1Cl N(C(=NCCCF)NCc1ccc(N2CCCCC2)cc1)CCNC(=O)C1CC1 Cc1nc2ccc(C(N3CCC(=CCNC(C4(C)CC4C)=O)CC3)=O)cc2[nH]1 O=C(CCCCC(F)F)NC1CCCN(C(c2nnn3c2CSCC3)=O)C1 C1(NC(C(C(C)C)SCC)=O)C2CC3CN(C(=O)CCN(C)CCO)C1C3C2 C1(CNC(=O)NCC(c2ccccc2Cl)N(C)C)CC2(CCOCC2)CO1 CC1(C)C2CCC1(C(N1CCC(CNC(=O)CC34CC(C3)C4)CC1)=O)C(=O)C2 Cc1cc(CC2CCCN(N3CCCCC3)C2)oc1.c1(C=O)ncn(C(C)C)n1 c1(C(=O)NC2CCN(C(COCC#C)=O)C2C)cc2c(C)ccc(F)c2[nH]1 c1(C(=O)NC(CC=C)(C)C)ccc2cc(Cl)ccc2c1 c1(C2C(C(N3CC(C)(NC(COCCCC#C)=O)C3)=O)C2)cccc(F)c1 C1(C(=O)NCC(C)N(C)C(c2ccc(C#N)cn2)=O)CCC2CC2CC1 S(=O)(=O)(c1ccc(Br)s1)NC1CCC(NCc2cc(C)c(Cl)cc2)C1 CC1CN(C(C2CC2(C)C(F)F)=O)CCN(C(=O)C(O)CC[S+](C)C)C1 c1(CNC(c2n[nH]c(C)c2Cl)=O)ccnc(O)c1F CC1=NS(=O)(=O)NC=C1C(=O)N1CCN(C(=O)CN2CCCNC2=O)CCC1C c1(C(=O)NC(=O)C(=O)N(CCCN(C(=O)NC(C)(C)C)C)CCO)nonc1N C1(CC)(CC)CCCN(C(c2cnc(C(=O)NC)c(Br)c2)C(=O)NC)C1 S(=O)(=O)(c1cccc(NC2CCN(C3CC3)C2)n1)N1CCN(CC)C(C)C1 c1(C(=O)OC)ccc(CCOC(C2CC2(c2ccccc2)C)=O)cc1Cl CC(C)S(=O)(=O)c1ccccc1CCC(=O)NC1CC(N2CCCC2)C1 C1(NC(C(CC(C)C)OC)=O)CN(C(c2nc[nH]c3ncnc2-3)=O)CC(C)(C)C1 C(CCCC(=O)OC(C)(C)C)NC(C1CC(C(C)(C)C(N)=O)C1)=O C1(N(C(c2nc(C)[nH]n2)C)C)CCCN(C(=O)Nc2ccc(OCCF)cc2)C1 CC(C)(C)C(O)C(=O)NCC1CN(C(C2(c3ccc(Cl)cc3)CC2)=O)CCCO1 C12(NC(CCC#CC)=O)CCCN(C(c3cccnc3C)=O)C1C2 C(N=c1cc(CNN2CC(C)(CC)OCC2)nc(C)[nH]1)c1c(C)cccn1.SC C1(C(=O)N(CC2(F)CC(NC(C(C)(C)NC(=O)OC)=O)C2)C2CC2)CC2CCC(C1)O2 C(CC1CCCC1)(C(=O)NC1CCC(C(N2CC(N(C)CCO)C2)=O)C1)OC N1(C(c2c(C)cccc2F)=O)CC2CC(NC(C3(C)CC3(F)F)=O)CC(C2)C1 c1(C(N2C(CNC(C(C)N(C)C)=O)CC2)=O)cc(C(F)F)cnc1O.C(C=O)SCC c1(C(N2C(CNC(C3Cc4ccncc4C3)=O)C=CC2)=O)cnn2c1NCCC2 N1(C(C)=O)CCCC(NC(=O)C(=O)NCC2CC2)C1 c1(C(N2CC(CSC)C2)=O)ccoc1CNC(=O)COC1CCCOC1 c1(NC(C(=O)NC(C)CC2CCCOC2)=O)cc(S(N)(=O)=O)co1 C1(NC(C2CCN(C(C3CC(O)C(F)C3)=O)CC2O)=O)C2CCC3C(C2)CC13 c1(NC(C)=O)ccc(OCCN(C(c2ccc(C(=O)OC)[nH]2)=O)C(C)C)cc1 N1(C(C2(CCN(C)C)CC2)=O)CCC(C(=O)NC2CCN(C3CC3)C2)CC1(C)C CCCC(CC)CC(=O)NCCC(C)NC(=O)C#CC1CCC1 C=CCC(CNC(=O)CC1CC=CCC1)C(=O)N(C1CCC1)CCO C1(CNC(c2cnc(NC)s2)=O)(NC(c2cncc(C)c2Cl)=O)CCCCC1C C(=O)(C(C#N)C(C)(C)C)NC(CCCC)CNC(=O)CCSC C(=O)(C(C)CC(C)(F)F)N(CCCCCCNC(c1c(C(C)C)c[nH]n1)=O)C N(C(=NCc1cc(C2CC2)[nH]n1)NC1CCCC1)CC(NOC)=O N1(C(c2nc(Br)nn2CC)C(=O)NCC)CCn2c(C)nnc2C1CCC C1(C(N2CCC(CCCC)C2)=O)CC2(CC(NC(=O)C=C3CCC3)C2)C1 c1(C(N2CC(NC(c3cc(C)[nH]c3)=O)C(C)CC2)=O)cccn2cncc12 C(=O)(CP(C)(C)=O)NCc1cn(C2CN(C(CN(C)C(=O)C3CC3)=O)C2)nn1 Cc1nccc(C(=O)NCC2CCN(C(C3CN(C4CCCCC4)C3)=O)C2)c1Cl c1(C(c2nnnn2Cc2cccs2)(C2CC2)NC(C=C)(C)C)ccc(Cl)cc1 C(CC1CC1)(CC(=O)NC(c1cnc(C)s1)C)NC(C1C(CC)CCO1)=O n1(CC)nccc1C(=O)NC1(CNC(c2csc(Br)n2)=O)CC1 N1(C(Cn2ccc(C)n2)=O)CC(C(=O)NC2CC=CCC2(C)C)CC1(C)C C1(NC(C(CNC(CC(=O)N(C)C)=O)O)=O)CC2CCC(C1)C2 c1(C(=O)OCC(c2ccc(C(CCC(=O)N(C)C)=O)cc2)=O)cc2cccnn2n1 c1(C(=O)NC(CNC(c2n[nH]c(C)c2Cl)=O)C)ccc(Br)cc1C#N c1(OC)ccc(Br)c(C(=O)NC2CCCC(NC(=O)C(C)OC(C)(C)C)C2)c1 C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)N1CCN(Cc2cnc(C)n2C(C)C)CC1 C1(O)(COC)CCCN(C(c2cc(CCNC(CSCC)=O)c(C)s2)=O)C1 NC1CC2CCC1CC2C(N1CCCc2n[nH]cc21)=O C(=O)(C(CC(C)C)C(N)=O)NC1CC2(CN(C(c3c(C)cc(Cl)cc3)=O)C2)C1 C12(NC(c3nn(CC)c(C)c3)=O)CCCC1N(Cc1cc(C)ccc1C)CC2 c1(C(=O)NC2(C)CC(NC(C(c3ccccc3)OC)=O)C2)ccc(CO)c(F)c1 CCC(C)C(O)C(C)C(=O)N1CCCC12CCN(C(c1cc(Cl)ccc1N)=O)C2 Brc1cc(=NC2CCNC3(CCC3)C2)[nH]c(NCc2c[nH]c3ccncc23)n1 C1(C(C(=O)N(CC(CC)NC(=O)CCOC(C)=O)C)F)CCOCC1 c1(C(=O)NCC2C(NC(c3c(C)cc(=N)[nH]c3)=O)C2)cc(C)n(NC(N)=O)c1C CCC(C)C(C(=O)NC1C=CC(CNC(c2ccc(N)cn2)=O)C1)OC C1(CC(=O)NC(c2ccc(O)cc2)=O)CC2(CCN(CC3C(C)C3)CC2)C1 C1(CCC)CN(C(=O)CC2CCCCC2C)CC1C(=O)NCCC(F)=C(F)F C1(CS(C)(=O)=O)CCCN(C(c2ccccc2F)=O)C1 c1(NCCC)ncccc1S(=O)(=O)NC(c1ccc(Br)cc1)C(C)C C1(CC(=O)N(C2CCSC2)C)CCCCN1C(=O)Cn1c(O)nnc1O N1(C(c2ccc(C#C)cc2)=O)CC(C(=O)NC(C)C)Cc2ccccc21 C1(CN(C(CC=CC=C)=O)C)CN(C(=O)C=CCO)CCO1 Cc1n[nH]c(C)c1CC(=O)NC(C1CN(C(c2cc(C#N)on2)=O)C1)C c1(CNC(N2CC(N(C(c3c(C(C)C)ocn3)=O)C)C2)=O)scc2c1OCCO2 c1(C(=O)NC2CCC(NC(CC(=O)OCC)=O)CC2)csc2cccc(OC)c12 c1(C(=O)NC2(CCNC(c3cc(OC)ncc3)=O)CC2)ccc(P(C)(C)=O)s1 Cn1cncc1CCC(=O)NC1C=CC(CNC(c2ccc(C(F)(F)F)s2)=O)C1 N1(C(c2n(C)cnc2)=O)CC(NC(C2CCCCC(=O)N2)=O)C(S(C)(=O)=O)C1 C(CC(C)C(=O)NCC#CC(=O)NCc1nc(C)sc1C)=CC c1(CC2CCN(C(C(=O)NCc3nnn(C)n3)=O)CC2)cnc(C(C)(C)C)nc1 N1(C(C2CCC(CNC(c3cccc(C)c3N)=O)O2)=O)CCOC(C)(C)CC1 CCC(CC(=O)N1CCC(C)(C(=O)NCC(F)CO)C1)C(C)C CCCC(CC)CC(=O)NC1CN(C(=O)CCC=C(C)C)CC12CC2 C(=O)(C(C(C)(C)C)NC(C)=O)N1C(CNC(C=CSC)=O)CCC1 N1(C(C2CCN(C(N)=O)CC2)=O)CCCN(C(c2ccncn2)=O)CC1CO N1(C(c2n[nH]c(C)c2O)=O)CCC2(CCCN(C(C3CCC(F)C3)=O)C2)C1 Cc1ccc(C(=O)NC2(CNC(C3CCCCS3(=O)=O)=O)CCC2)cc1C c1(C(=O)NCc2cn(C3CC(C(=O)OC)C3)nn2)c(C)nc2cccnn12 c1(N2CCC(C)C2)ccc(C(=O)NC2(CNC(=O)C=CCF)CCOC2)cc1 C1(CC=C)(C(N2CCCCC2CNC(c2ccncc2C)=O)=O)CCOCC1 CCC(C)CC(=O)N1CC(CC(C)NC(c2cnn(-c3ccccc3)c2Cl)=O)C1 c1(C(N(C2CCN(C(CCC(C)OCC)=O)C2)C)=O)cccc(Cl)c1N c1(C(=O)NCCC(=C)CC(=O)NC2CC2c2cccs2)ccnc(CO)c1 c1(OCc2nc(C)sc2)cccc(Cl)c1Cl.c12cn(nn1)CC1CCCN1C2=O Cc1cc(C(N2CCC2CC(=O)NCC(C)C#N)=O)c[nH]1 c1(C(=O)NC(CC=C)CNC(C2CC3CC3C2)=O)c(N)c(C(F)(F)F)nn1C c1(N2CC(C)=C(C)CC2)[nH]c(=NCC2(CO)CC=CC2)nc2sccc12 CC1CN(C(c2ncnn2C2CC2)=O)CC1CNC(C1CS(=O)C1)=O C1(OC)CCCCC1C(=O)NC1CCN(C(=O)CN(c2ccc(Cl)cn2)C)C1 CC(CC(F)F)C(=O)NC1C2CC1N(C(C1C(F)(F)C13CCC3)=O)C2 c1(C(=O)NC(C2CCN(C(C(C=C)(C)C)=O)CC2)C)c(N)sc2c1CCSC2 c1(C(N(CCC(C)NC(=O)CN=S(C)(C)=O)C)=O)cccc2cncn12 c1(SCC)cccc(C(=O)NCCC2CCCN2C(=O)Cc2cc(C)no2)c1 c1(C(=O)NCC(CN(C)C(C2CC(N(C)C)C2)=O)(C)C)cc2cc(Cl)ccc2[nH]1 c1(NC2CCN(C(C(CC)OC)=O)C2)ncnc(Cl)c1C(=O)OC N1(C(Cn2cc(-c3onc(C)n3)nc2)=O)CCCC2(CCN(C)C2=O)C1 N1(C(C2CC(NC(CCOC(C)=O)=O)C2)=O)CCCC(C(F)(F)F)C1 C(=O)(CCC(=O)c1ccccc1Cl)N1C(CNC(C2(CC)CC2)=O)C=CC1 N1(C(C(C(C)C)(C)O)=O)CCCCC2(C1)CN(C(c1cccc(S(C)=O)c1)=O)C2 c1(CC(=O)NC2CN(C(c3ncn(CC)c3)=O)C2)cccc2cnccc12 C1(NC(c2ccnc(OC)n2)=O)CCC2CN(C(=O)CS(=O)(=O)N(C)C)CC2C1 Cc1c(NC2CCCS(=O)(=O)C2)ncnc1N1CCCC(CC(F)F)C1 CN1CC(O)(CN(C(=O)CCC2(C)CN(C(=O)C=C3CCCCC3)C2)C)C1 c1(CCC(=O)Nc2c(OC)ccc(OC)c2)cccc(S(=O)(=O)N(CC#N)CC)c1 N1(C(C(=O)NC(CC)(C)C)CCc2ccsc2)C(CO)CC2OC(C)CC12 c1(CN=c2scc(C(N3CCC(O)C(F)C3)=O)[nH]2)ccc(F)c2ccoc12 C12(NC(CCCc3ccc(C)cc3)=O)CCC(NC(=O)Cc3ccno3)(CC1)C2 C1(NC(CNC(C2C(C)C2)=O)=O)CC2(C1)CC2NC(=O)CN(CC(C)(C)C)C c1(NC(C2CC2NCc2ccc(-n3ccnn3)cc2)=O)cccc(F)c1CO S(=O)(=O)(c1ccc(NCc2ccnc(N(C)C)c2)nc1)NCC=C=C c1(C(C(=O)NC(C)(C)C)N(C)Cc2ccc(Cl)s2)ccc2c(c1)C(=O)N(C)C2 C1(NC(CCN2CCN(C)CC2)=O)CCC2CN(C(=O)C3=CCSC3)CCC2C1 CCCCC(C(=O)NCC(C)(C)OCC(=O)Nc1ccc(F)cc1OC)C(C)C C(=O)(C(C)C(=O)NCc1ccc(C(=O)N(C)Cc2cocn2)o1)OC n1(CCC(=O)N(C2CC(NC(C3CCC3CF)=O)C2)CC)cnc2ccccc12 CC1CC(CNC(=O)CC2CCCC2NC(C2(N(C)C)CC2)=O)=NO1 C=CCC(C)(C)CC(=O)NCCC1C(C)CCCN1C(=O)CNC(=O)OC c1(C(=O)NC2CN(C(CC(CCC)C)=O)C(C)CC2)cn(C)c(=O)nc1O N1(CCCC(=O)NC(CCC(C)C(=O)O)=O)CCc2ccccc21 N1(C(c2c(OC)c[nH]n2)=O)CC2CN(C(c3c(C(F)F)n[nH]c3C)=O)CC2C1 C(CN=C(NCC(c1cccnc1)O)NCC1CC1)c1ncc(C)s1 c1(CC(=O)NC2C(C)(C)C(CNC(=O)COc3ccccc3)C2)cc(F)ccc1Cl c1(CC)oc(C(=O)NC2CCOC(C(=O)N(C)CCN(C)C(C)=O)C2)cc1C c1(C(=O)NCCC2CCCN(C3CCN(C)C3=O)C2)ccc2c(c1)C(=O)NC2 CN1CCCCC(NC(=O)CC(CC2CC2)NC(=O)C(O)c2ccco2)C1 N1(C(c2cccc(C)c2)=O)CCC(NC(c2c[nH]c(=O)cn2)=O)C2(CCC2)C1 C(=O)(CCS(C)(=O)=O)N(CCNC(C(C)=NOCC#N)=O)C Cc1cc(F)cnc1C(N1CCC(NC(=O)CN2CCCCCC2)C1C)=O c1(OC)ccc(C2(NC(=O)C(N3CCN(C(=O)CC#N)CC3)C)CC2)cc1OC C1(CNC(C(C)OCC#C)=O)CC2CCC(C1)N2C(=O)CC1(OC(C)=O)CCCC1 C=CC1OCCC1C(N1CCC(N(C)C(c2ccc(OC)cc2)=O)C1)=O C(=O)(C1=NOC(C2(O)COC2)C1)N1CC(CCNC(=O)CC2CCC2)C1 Cc1cc(F)ccc1C(N1CCC(NC(=O)CCn2ccnn2)C1C(C)(C)C)=O C1(C(C)C)(C(=O)N(C)Cc2ccon2)CCCN1C(=O)C(N1CCOC1=O)C C1(NC(=O)CCOCCCNC(=O)CC2CCCSC2)(CO)CCSC1 c1(C(=O)NCC(CN(C(=O)Cc2nc[nH]n2)CC)(C)C)cccc(C#CCO)c1 C(=O)(C1=CCCCO1)N1C(CC(=O)NCC2CCC(C)CC2)CC(O)C1 c1(C(=O)NCCN(C(C2CC=CCO2)=O)CC)cnc(CC(C)C)s1 C12(C(=O)O)CCCC1CCN2C(C)=O.C1(C(N(C)CC)=O)CC1C(F)F Cc1cccc2c(C(=O)N(C)CCNC3(C4CC4)CCOCC3)coc12 CCC(F)(F)C(C)(C)CN=c1cc(C)[nH]c(=NCCCC2CC2C)[nH]1 Cc1ccc(C(=O)NC(CNC(=O)CN(S(C)(=O)=O)C)CC(C)C)c([N+](=O)[O-])c1 Nc1c(C(=O)NCCOCCCNC(C2CCC(F)(F)C2)=O)ccc(F)c1F CCCC(C(=O)N1CC(O)CC1C(=O)NCc1conc1COC)OC c1(C(N2CC(C)(c3cn(-c4cccc(Cl)c4Cl)nn3)C2)=O)c(Br)cccc1Br c1(OC)cc(Cl)c(CNC(=O)CC2COCC3(CCC3)O2)cc1OC c1(OC)ccc(F)c(N)c1C(=O)N(C1CCCCC1N(C)C(=O)OC(C)(C)C)C Cc1c(C(=O)NCC2(NC(c3cc(N(C)C)nc(Cl)c3)=O)CCC2)cccc1N N#CCCCC(=O)N1CCC(OCCNC(=O)C(F)(F)CF)C1 c1(C(C)C)ccccc1-n1nc(CC2CCC2)nc1-c1ccsc1Br C(=O)(CC(C)C(C)(C)C)N1CCCCC(CNC(c2c(COC)scc2)=O)C1 C(C(C)(C)NC(=O)CC1CCCO1)=CC(=O)N(C)CC1CCSC1 C(=O)(C1CCCc2scnc21)NC12C(CN(C(CCOC)=O)C1)CCC2 CCCC(C)(CCC)C(=O)NCC(C)NC(c1[nH]cc2c1CCCC2)=O C1(NC(C=COCC)=O)CN(C(=O)CN2CCC(O)CC2)C(C)(COC)C1 C1(NC(c2c(CC)nco2)=O)CCC2CC1CN2C(c1cnc(C(C)(C)C)s1)=O Cc1cc(C(=O)N(C)CC2CN(C(C3CC(C)(C)C3)=O)CCO2)c(C)n1C1CC1 C1(C(N(CCNC(C(c2c(F)cccc2F)C)=O)C)=O)CCC2(CCC2)C1 c1(CN(C(C)CS(C)(=O)=O)C)ccc(C#N)cc1Br c1(C(N2CC(NC(C(CC)C(C)C)=O)C(C)C2)=O)cc(F)cc2ccoc12 CC1C(NC(=O)CC2(C)CC2)CC2CCC1N2C(=O)CCCC(=O)C1CC1 c1(-n2cnc(C(=O)NCCN(C(C(CC)OCC)=O)C)n2)ncccc1F C1(C)(C(=O)NCC2C(CNC(c3c(C(C)=O)coc3)=O)C2)CC=CCO1 N1(C(c2cc(C3CCC3)on2)C(=O)NCC)CCC2(CCC(O)C2)C1 CN1CCCCC1C(=O)NC1CCN(c2nnc(-c3ccon3)s2)C1 CC1CN(C(C2(C3CCC3)CC2(F)F)=O)CC(C)N(C(=O)CCS(C)=O)C1 Cc1ccc(-c2ccc(F)c(C)c2Cl)c(C#N)c1 Cc1nc(C)c(C(=O)N(CCCNC(c2cc(Br)sn2)=O)C(C)C)o1 C1(CNC(c2c[nH]nc2C2CCCCC2)=O)CC(O)CN1C(=O)CCCF C1(C2CCN(C(=O)CC3CCCOCC3)C2)(NC(C(C(C)C)CO)=O)CC1 C1(CNC(C(CC)COC)=O)CN(C(=O)CCc2cc[nH]n2)CC12CCC2 C(C(=O)NNC(=O)c1ncccc1Br)Oc1c(C)cccc1.c12noc(n1)C2 NC1=CCC1CNC(=O)NCC(=O)NC(CO)C1(O)CC1 C=CC(O)(C(=O)N1CC(NC(=O)CN2CCCCCCC2=O)C(O)C1)C(F)(F)F C(=O)(CCCN(C)N=O)N(CCCNC(C(C(CC)O)C)=O)CC1CCCC1 N1(C(C(C)Cc2cccc(Br)c2)=O)CC(NC(c2c(Cl)cnn2C)=O)C(C)C1 N1(C(C(C)Cc2cccc(F)c2)=O)CCCC(O)(CNC(=O)COC2CC2)CC1 CCC(CC)CC(=O)NC1CN(C(=O)C(C)(C)C2CCCCO2)CCC1C C1(CN(C(c2coc(-c3ccc(OC)cc3)n2)C(=O)NC)CC=C)CCC(C)(C)C1 N1(C(CCCC=C)=O)CC2(CCCC(CNC(=O)C(C)(C)N(C)C)O2)C1 C1(C)(CNC(C(C)NC(=O)NC)=O)CCN(C(=O)COc2ccccn2)CC1 CCCCC(C(=O)N(CC(C)NC(c1ccnc2cc[nH]c12)=O)CC)C(C)C S(=O)(=O)(c1ccnn1C1CCOCC1)C1CCC(C)C(CC)O1 C1(C(N(C(C)C)C)=O)CC2CCC(C1)N2C(C1CC(O)C1)=O N1(C(=O)COC2(Br)CC2(F)F)CCC(O)(c2noc(-c3ccccc3)n2)CC1 C1(CC(=O)NC2(CCNC(c3c(OCC)cccn3)=O)CC2)OCCOC1(C)C CC1CCC(C(=O)Nc2cnn(-c3ccccc3)c2)N1C(C1CCC(=O)N1)=O C1(C)(C(=O)NCCc2onc(C)n2)CC12CCN(CC(=O)NCC1CC1)CC2 C=CC(CC)CC(=O)NCC1CN(C(C2(C)CCCCNC2=O)=O)CC1(C)C Cc1cc(C(N2CCCC2Cn2cc(C3CC3)nn2)=O)c2c(C)n[nH]c2n1 c1(N)noc(CNC(C(=O)C2(C)CC2)=O)n1.c1(CCS)csc(-c2ccccc2)n1 Cc1ccc(O)cc1C(=O)NCCC1(O)CCN(C(=O)CCC2CC2(F)F)CC1 CC1CCc2[nH]nc(C(=O)NCC3(CNC(C4CCOC(=O)CC4)=O)CC3)c2C1 C1(C(=O)NCC(CC)N(C)C(c2cc(C3CC3)nnc2O)=O)CCCCCCC1 C1(C(N(CC(=O)OC)C)=O)CN(C(=O)C(C)CSC)CC1(C)C c1(C(N2CCC(NC(CC(=C)C)=O)C(C)C2)=O)nc(C(F)(F)F)n2c1CCCC2 C1(CNC(CCN(C)CCc2cc(F)ccc2F)=O)CC2(C1)CC(C(F)(F)F)C2 c1(N2CCC(C)(OC)C2)ccncc1S(=O)(=O)N1CCCC1CCO C=CCCCC(C)(C)C(=O)NC(C)CC(C)NC(=O)CCc1nccn1CC N1(C(C(C=C)(C)CC)=O)CCc2ccc(C(N3CCOC(C)C3C)=O)nc2C1 c1(C=O)cnc2c(c1)COCC2.C(=O)(CC(=O)N)NCCCN(C)N(C)CC1CC1 C12(NC(=O)COC3CCOCC3)CC1CN(C(c1ccccc1C(F)F)=O)C2 c1(C(=O)NCC(C(N2CCC(C)C2)=O)N(C)C)cnc(O)c(Cl)c1 CCC(C)(CNC(C1CCCN1C(=O)Cn1ccnc1)=O)C(N)=O C(=O)(CC(CCC)CCC)N1C(C(=O)NCCSCC=C)C(C)C1 N1(C(C(CSC)OC)=O)CCC2(CC(NC(c3nnn(C)n3)=O)C2)C1 C1(c2cn(C3CC(C(=O)NCCc4n(CC)cnn4)C3)nn2)CCN(C)C1=O C1(CC=C)(C(=O)NCC2C=CCCC2)CCN(C(c2cc(C(C)C)on2)=O)C1 C12=NC(=N)NC(=NCCCN1)N2.CC1CS(=O)(=O)CC1N(C)CCO N1(C(C=C(C)C(F)F)=O)CC(CNC(=O)CNc2nccs2)CC1(C)C C1(C2CCC2)(C(N2CCN(C(COCC(=O)NC)=O)C(CCO)C2)=O)CC1(F)F c1(C(=O)NCCCN(C(=O)CC2CCC2(C)C)C)cc2cc(Cl)ccc2n1C c1(N2CC3C(NC(C(CC)(C)C)=O)(C3)C2)ncc2ccsc2n1 C1(NC(=O)CCC2CCCC2)CCN(C(C23CCCC(C2)OC3)=O)CC1F CN1CCC(F)(C(=O)NCCCNC(=O)C=CC(c2ccc(F)cc2)=O)CC1 N(C(=NCCOc1ccc(C(C)C)cc1)NC1CC1C(F)(F)F)CC N1(C(c2n(CC(C)C)ncc2)=O)CCC(O)(C(C)NC(=O)C(C)CCF)CC1 C1(C(=O)NC2(C(=O)NCCCCCOC)CCN(C)C2)CCC(N=[N+]=[N-])C1 c1(C(=O)NCCCOCCNC(C(C2CCC(=O)N2)C)=O)cccc(N)c1F C(=O)(CCCC(C)(C)N(C(C)CN1CCCC1=O)C(C)=O)NCCCC N1(CC(=O)NC)C2CCC1CC(NC(C1CCC(C)C(C)C1)=O)C2 c1(-c2c(OC)nccc2)ccc2oc(C(=O)N=c3[nH]nc(C)o3)cc2c1 c1(CC)ncc(C(N2CC(CNC(C3CCOC3C)=O)C2)=O)c(C)n1 CN1CCOC(C(=O)NC2CC(F)CN(C(c3cc(C4(C)CC4)on3)=O)C2)C1=O c1(C(N(CC(C)NC(=O)CC2CC(=O)NC2=O)C)=O)ccc(C(F)(F)F)c(F)c1 N1(C(C(C)C2CCCC2)C(=O)NC2(C)CC2)CCC2C1CC1(CCC1)C2 N1(C(C2(C)C=CCC2)=O)CCCC2(NC(=O)C(F)=CC3CC3)CC2C1 c1(C(N2CC(C)C(NC(C3CCCC(F)(F)C3)=O)C2)=O)cc(O)cc(=O)o1 c1(C(=O)NC2C(NC(C3(CCOC)CC3)=O)C2)cn(C(C)C)nn1 c1(OC)ccccc1SCC(=O)NC1CC1CNC(=O)C(c1ccc(C)s1)C.COC CCC1=C(C(=O)N2CCC(C(C)NC(c3cnn(C)c3)=O)C2)SCCO1 C1(C(N(CC)Cc2ncsc2NC)=O)CCCN1C(=O)C(C1CCOCC1)F C1(C(=O)NCCCN(C(C(C(C)C)c2cnn(C)c2)=O)C)CCn2nccc2C1 C1(C(=O)NCC(C(C)(C)O)(F)F)C(C2CC2)CCN1C(=O)C=Cc1nccs1 c1(NC2C(C)CCNC2)ncnc2sc3c(c12)CCC3.c1(CC=O)ccoc1 C1(CC=C)(NC(=O)CC2CCCO2)CCN(C(C2(C#N)CC2)=O)C1 C(=O)(CCS(=O)(=O)N(C)C)NC1CCC(N(C(CCC=CC)=O)C)C1 N1(C(CCCN(C)C)=O)CC(O)CC1CNC(C1CC1C(C)(F)F)=O CC1(C)COCCC1NC(C1CCCN1C(c1ccc(F)nc1F)=O)=O C12(CC(=O)NCCOC3CCN(C(c4c[nH]nc4Cl)=O)C3)CCCC1C2 c1(CC)cccc(C(N2CC(CNC(c3cc(SC)c(C)o3)=O)C(C)C2)=O)c1N C(=O)(CC1CCC(=O)c2ccccc21)NC1CC(C)(N2CCOCC2)C1 N1(C(C(C)CN(C)C)=O)CC(O)(C2(CNC(=O)CC3CCC34CCC4)CC2)C1 C1(CC(=O)NC(c2ccccc2)C(C)NC(c2c(C)scn2)=O)CCCC(=O)N1 N1(C(c2cc(CC)sn2)=O)CCOCC1CNC(c1cnc(C(C)(F)F)s1)=O C=CCC(CNC(C1CCSCC1)=O)C(=O)NCc1nnc(O)n1C N1(C(c2c(C)onc2C2CC2)=O)CC2(C1)CN(C(=O)CC1CCCCC1O)C2 CC1(CNC(C2(C)CCCO2)=O)CCCN(C(=O)C=Cc2ccncn2)C1 c1(C(=O)NCC2C(NC(CNS(C)(=O)=O)=O)C2)ccc(C2CCC2)cc1 C(C1(C)COC1)=CC(=O)N(CCOCCN(C)C(C12CCCC1C2)=O)CCO c1(CCN=C(NCC2CC(C)OCC2)NCC2CCC2)ccc2ncccc2c1 CCC(C)CCC(=O)NC1CCCCN(C(=O)CCOCCCOC)C1 N1(C(CSCCC(C)C)=O)CCCCC1CCNC(=O)C=Cc1ccn(C)c1 c1(C(C)(O)C(=O)OCC(=O)Nc2ccnn2CC2CCCO2)cccc(Br)c1 c1(C(=O)NCC(CC)NC(=O)Cc2ccno2)cc(O)cc(Cl)c1Cl C(C(C)C)(C(O)C(=O)N(CCCCCNC(=O)CN1CSCC1=O)C)OC c1(C(=O)NCC(CNC(C(=O)NC)=O)F)cc(F)c(F)cc1NC(=O)C1CC1 CC1(C)CN(C(C2CC(CF)C2)=O)CC(CNC(C2CNC(=O)N2)=O)O1 C1(CNC(C2(C(CC)=O)CC2)=O)CCN(C(C2CCN(c3nc(=N)[nH][nH]3)C2)=O)C1 CC1(C)CC(=O)N(CC(N2CCCC2CNC(c2c[nH]nc2C(F)F)=O)=O)O1 N1(C(C(C)OCC#C)=O)CC(C)(CNC(=O)CNS(C)(=O)=O)CC1(C)C C1(C(=O)NCC(CC(=O)NCC(C)N(CC)CC)O)Cc2nccn2C1 n1(CC(=O)NCC(C)CN(C)C(c2cn(C)nc2O)=O)sc2ccccc2c1=O CC(CCNC(C1(C(C)NC(C2CCCN2C)=O)CC1)=O)CCO C1(O)(CN(C(COCCCOC)=O)C)CCCN(C(=O)CCc2cnc(C)o2)C1 Cc1ccc(OC(C)C(N2CC(O)(CNC(=O)CCCSC(C)(C)C)C2)=O)cc1 C(=O)(CS(=O)(=O)C1CC1)N1CC(CN2CCN(C(C34OC(C)C(C3)C4)=O)CC2)C1 N1(C(C2(C)CN(C(c3ccc(CO)nc3)=O)C2)=O)CCCC(C(N)=O)CC1 CCC(CC)C(F)C(=O)N1CCN(C)C(CC(=O)NCC2CC(=C3CCC3)C2)C1 C1(OC)CC(C(=O)NCCCNC(C)=O)N(C(C2CC2C)=O)C1 c1(CN(CC=C)C(C2CCN(CC3CCOC3)CC2)=O)cc(Br)ccc1F C(=O)(C1CCCc2ncnn21)NC1CN(C(c2cc(N)nc(Cl)c2)=O)CC12CC2 c1(C(N2C(C(=O)NCC(N)=O)CC(O)C2)=O)c[nH]c2nccc(Cl)c12 CC(CC(=O)N1CCC(n2ccnc2)C1)C(C)(C)NC(c1cc(C(N)=O)co1)=O C1(N(C(C(C(C)NC(=O)CCc2nc(=N)[nH][nH]2)C)=O)C)CCCC(C)(C)C1 N1(C(C(CC)C(=O)OC)=O)CCN(C(=O)CCOc2ccccc2)CC(O)C1 C1(CC(=O)OC)CCC2CN(C(=O)Nc3ccc(C4CNC(=O)C4)cc3)CCC2C1 C(=O)(C(C(C)O)NC(C1CCNC1=O)=O)NC(C)Cc1ccco1 C1(NC(c2c(C)cccn2)=O)CC2(C1)CC(C(=O)NC1CCOC(C)C1)C2 Cc1nc(N(CCCCN(C)C(c2cn[nH]c2)=O)C)c2cc[nH]c2n1 C1(NC(C(=O)NCC2C(CC)CCCC2)=O)CCCCC12CC2 C(=O)(C1=CCOCC1)N(C(C(=O)N(C(C1CCOCC1)C)C)c1ccoc1)C1CC1 C1(CNN(C(C)(C)C)C(=O)CC2(NC3CC3)CCC2)CC2CC2C1 C1(CNc2ccc(C(=O)Nc3snc(CCC)n3)cc2)CC(F)CN1C(N)=O N1(C(C2C(C)(C)CO2)=O)CC2CC(NC(c3ccc4ccnn4c3)=O)CC2C1 N1(C(C2CC=C(C)CC2)=O)CCC2C1CCN2C(C1CCCSC1)=O N1(NC(C2N(C(C(c3ccc(OC)cc3)C)=O)CC(C)C2)=O)CCC(F)(F)CC1 C1(C)(CC)CC(NC(=O)CN(C)CCOC)CN1C(C1COCCN1C=O)=O Cc1cc(C(=O)NCC2CCOC2C)nn1CCO c1(C(N(C2CCC(NC(=O)C(C)SC)C2)C(C)(C)CC)=O)sccc1OC(F)F C(Cn1cncn1)(C(=O)NCC1CCC(NC(=O)CCCc2cncs2)C1)OC NS(=O)(=O)c1ccc(OCC(N2CCCC(NC(=O)Cc3cnc[nH]3)C2)=O)cc1 C1(CCN(C(c2cn(CC)nc2)=O)C)CCN(C(c2ccc(OC)s2)=O)CC1 C12(C(=O)NCC3CCN(C(C4(C)CC=C(C)CC4)=O)C3)CCCN(CCC1)C2 N1(C(C(C)NC=O)=O)CC(NC(=O)CCc2ccc(N)cc2)C(C)(C)C1 CC(O)(CC(=O)NC12CC(CNC(c3sccc3CC#N)=O)(C1)C2)C1CC1 CC(C)C(C)C(=O)NCC12CC(NC(=O)CC3CCCC4CC34)(C1)C2 C#Cc1ccc(C(N2CCC(CNC(c3cscn3)=O)CC2)=O)c(F)c1 c1(C(=O)NC(C2CN(C(=O)CO)CCO2)C)ccn(CCO)c(=O)c1.C1NC1 c1(C(=O)NCC2N(C(C(=O)NCC)=O)CCN(C)C2)cc2ccccc2c(=O)o1 C12(C(=O)NCC=CC(=O)NC(C)CS(C)=O)CC1CNC2=O S(=O)(=O)(c1ccc(F)c(C)n1)NC(c1ccccc1CSC(F)(F)F)CC N1(C(C(CCC)OC)=O)CCOCC(F)(CNC(c2cc(C)[nH]n2)=O)C1 C1(NC(CC(CNC(C2(CC#C)CCCO2)=O)O)=O)CCC(C2CC2)C1 c1(N2CC3CC(NC(C=C(C)C)=O)C3C2)nnc2c(c1C#N)CCCC2 c1(C(=O)NCC2CC(C)N(c3nccc(C(C)(C)C)n3)C2)cnc2n1CCCC2 C(CC(=O)NC1(OCCNC(COCC)=O)CCCCC1)(C(F)F)OC C(CCC(C)C)(C(=O)NC1CCN(C(=O)C2=NNC(=O)CC2)C(C)C1)NC(C)=O C1(C(=O)NC(CC(C)C)CO)CCCC12CCN(Cc1cc(I)ccc1Br)C2 C1(NC(=O)CC2CC2C(F)(F)F)CN(C(=O)CCCn2cccc2)CCC1O N1(C(c2onc(CC)n2)=O)CC2(CC(NC(C3(C)CC=C(C)CC3)=O)CO2)C1 c1(C(N2C(C)C(NC(C3C4COCC34)=O)CCC2)=O)ccc2c(c1)OC(C)(C)O2 c1(Cn2c(-c3cccc(-c4cnc(C)c(Cl)c4)c3)ncc2)nc2cc(O)ccc2[nH]1 C(CCCCC(=O)NCc1ccc(C(=O)NCc2cnc(OC)cn2)nc1)=CC Cc1ccc(N2CCC2c2cn(Cc3nc(=O)o[nH]3)nn2)cn1 Cc1cc(Br)ccc1C(=O)NCC(CNC(C1(C)CC=CCO1)=O)CO C(C)(C)(CC(=O)N(C1CCC(NC(c2ccc(C(C)C)nc2)=O)C1)C)OC c1(CC)cc(OCC(=O)C2CCC2)ccc1Cl.C1C(C)CCC2(CC2)C(=O)N1 c1(N2CCCC(C(=O)N(CCCO)C)(CC)C2)ncnc2c1ncn2C(C)C1CC1 CC(C)C(C(=O)NC(C(N)=O)C1CCCC1)C(C)NC(c1ccc(CO)nc1)=O CC12CCN(CC1)CC2NC(C1(C)CN(C(c2cnsc2)=O)C(C)(C)C1)=O c1(C(=O)NCCOCCCNC(c2cc[nH]n2)=O)ccn2c(O)nnc2c1 N1(C(c2nc(CNC(=O)CCCC(C)=O)sc2)=O)CC(OCC)CC2(CCC2)C1 c1(CC(N2CCC(CCNC(C3(C#C)CCC3)=O)C2)=O)sc(C)nc1C C1(CNC(C(C)N=[N+]=[N-])=O)CC(O)C(O)CC1C(=O)NCCCCOC(C)C c1(C(=O)NCC(C)(CO)NC(c2cnn(C)c2F)=O)cn(CCO)c(=O)nc1O c1(C(=O)NCC(C)NC(C2CSCN2C)=O)cnc2c(c1)CCCC2 N1(C(=O)Cc2ccc(F)cc2Cl)CCC2C1CCN2C(C1(O)CC1)=O C(CC(C(=O)NCC)NC(=O)OC(C)(C)C)OCC=C.c12ncc(cn1)oc2=O N1(C(CC=CC=C)=O)Cc2[nH]nc(C(=O)Nc3cc(O)ccc3C)c2C1 Cc1occc(=O)c1C(N1CC2CC1CN2C(c1ccc(C2CC2)cc1)=O)=O Cc1nc(CO)ncc1C(N1CCCC(CCNC(C2CC2(C)Br)=O)C1)=O N1(C(=O)C2CC2)CCC(NC(CCN(C(C(C)OC)=O)C)=O)C1 c12ccc(cn1)C(=O)NC1CCCC1CN2C.C(=O)(C(F)(F)COC)NC.CCCO C(=O)(CCC(=O)N(C1CC(=O)N(CC2CC2)C1)C)NCCOCCCOC c1(CC)ccsc1C(=O)NC(C)C=CC(N1CCC(CC2CC2)C1)=O C(=O)(C(CNC(=O)C(O)C=C)CC=C)NC(CC#C)C(=O)NC c1(C(=O)NC2CC(NC(CC3CC(C)C3)=O)C2)cnn(CC2CCCCC2)c1C N1(C(c2cc(CNC(c3c(NC)scn3)=O)ncc2)=O)CCC(C)(CO)CC1 c1(N(C)CC2CN(C)C2)nc(=NCCC(C)(C)C)[nH]c2c1SCC2 C(c1ccc2c(c1)OCO2)=CC(=O)NCC(CNC(C(CC)(C)C)=O)CO c1(OC)cncnc1C(=O)NCC=CCNC(C12COC(C(F)(F)F)(C1)C2)=O N1(C(C(C(C)C)N(C)C)=O)CC2(CCN(C(c3cnc4n3CCC4)=O)C2)C1 N1(C(C2C(C)(C)CO2)=O)CCC2(CC1)CN(C(C1CCC(F)CC1)=O)CCO2 C=CCC(CC(F)F)C(=O)N(C)CC1CCCN(C(c2ccc(N)c(N)n2)=O)C1 c1(C(N2CCCC(NC(COC)=O)(COC)C2)=O)c(F)cc(C)cc1Br N1(C(CC2(C=C)CN(C(=O)CCc3ccncc3)C2)=O)CCOCCC1CC CCC(C#N)C(=O)N1CC(C(F)(F)F)C(CNC(c2ncc(C)cn2)=O)C1 N1(C(C2(OC)CCCOC2)=O)CC2CCOCC2(NC(=O)CCCCCOC)C1 c1(OC)ccnc(C(N2CCCC2CCNC(=O)CCC2CCCCO2)=O)c1F C(=O)(CCC(C)(C)C(=O)N1C2CCC1CC(NC(=O)C(C)C(C)O)C2)OC N1(C(C23CCC(OC)C2C3)=O)CC(NC(=O)CCSCC(N)=O)CCC1C c1(C(=O)NC2CN(C(COCCC)=O)C2)cn(-c2ccccc2)nn1 C1(C(N2C(C)(COC)CC2)=O)(C(C)C)CCN(C(c2cc(OC)n[nH]2)=O)C1 C(CCC(C)C)(C(=O)NCCC(C)CC)NC(C(C)OCCOC)=O C1(OC)CCN(C(c2cncc(CNC(C3SCC=C3C)=O)c2)=O)C(C)C1 C(=O)(CC(C)C(F)F)N(CCC(C)NC(c1c(C)oc(C(C)C)n1)=O)C c1(C(N2CCC(O)(C(=O)NCc3cccc(CO)c3)C2)=O)cccc(O)c1 C1(c2n(C(CC)(C)C)nnn2)(NCCCn2ccnc2CC)CC2CCN(C2)C1 CC1(C)CC1CC(=O)N(C(C(=O)NC1CC(n2ccnc2)C1)C1(C)CC1)C1CC1 C=C=CCCC(=O)N1CCCC(NC(C2(O)CCSCC2)=O)C1 Cc1c(C(=O)NC(C)CC(C)NC(C2CCCC23CCC3)=O)cccc1F c1(C(=O)NC2(C(N(OC)C)=O)CC2)cc(CNC(=O)CC2COCCO2)on1 Cc1cc(C)c(NC(=O)CCC2CN(C(=O)CC3CCC(=O)C3)CC2C)c(C)n1 Cc1nc(=NC2CC3CN(C(=O)CCc4cc(Cl)cs4)CC23)s[nH]1 CC(C)C(C(=O)N(C)CCNC(c1nc(C2CC2)oc1C)=O)C1CCC1 c1(OC)cc(C(N2C3CCC2CN(C(C2(C)CC2(F)Cl)=O)C3)=O)ccc1[N+](=O)[O-] C=CC1(C(=O)NCc2cccnc2Cl)CCN(C(C2CN(C(N)=O)C2)=O)CC1 CC(CCC(C)(C)C)C(=O)NC1CC(O)(CNC(c2n[nH]c3c2CCSC3)=O)C1 C1(C)(OCC)CCCN(C(C2CCCCCN2)=O)C1 CC1(NC(=O)CC2CCOC2=O)CCCCC1C(=O)NC1CC(O)CC1O C(CC(C(C)C)NC(c1c[nH]nc1F)=O)N(C(C1C(=C)C1)=O)C C#Cc1ccc(NC(=O)C(C2CCCO2)NC(c2scnc2CC)=O)cc1 C1(C(=O)NC2CCN(C(CCOC)=O)C2)CNC(=O)CC1(C)C CCCCC(O)C(=O)N1CCC1CNC(=O)Cn1ncc(Br)n1 N#Cc1cncc(C(=O)NC2C3CCC2N(C(C2CCN(C4CC4)CC2)=O)C3)c1 c1(C(=O)NC2(CC=C)CCN(C(C3CC3(C)C)=O)CC2)nncc2c1CCCC2 c1(NC(N2CCC(CNC(C(C(C)C)NC(C)=O)=O)C2)=O)cnc(O)c(C)c1 N1(C(c2csc3cncn23)=O)CCC2CCCN(C(=O)CC3CCCCC3)C2C1 C(=O)(C(CO)C(F)(F)F)NC(CC(N1CC(COC)OCC1)=O)C S(=O)(=O)(c1ccc2nc(N3CCCC(CCN(C)C)C3)sc2c1)NC(C)CC#N C1(C)(C(N2CCC(NC(C(CC)OC)=O)C(F)(F)CC2)=O)COc2ccccc2O1 N1(C(CCCOC(C)C)=O)CC(CNC(=O)Cn2cc(N)cn2)C(C)C1 N1(C(COC(CC)C)=O)CCCC(CC(=O)Nc2cccc(O)c2)C1 C12COC3(CCN(CC3)C1=O)C2.N1(NC(=O)COc2ccsc2)CCCC1CO c1(NC(CCCOC)C2CC2)nc(C)cc(=NCCCOCC(C)C)[nH]1 C(C)(CCC(=O)N1CC=CCO1)N(C(C(CCC)C(C)C)=O)C CC(C)C1=NOC(C(=O)NC2CC(O)C2CC(N2CC3(CO)CC3(CO)C2)=O)C1 C(CCCCC(=O)NC1CC12CC(O)C2)NC(=O)CC1(O)CCC1 c1(C(=O)NC2CCCCN(C(c3n[nH]c(=N)s3)=O)C2)cncc2c(F)cccc12 c1(C(=O)NC2CC(CSC)C2)ccnc(OCCNC(C(CC)OC)=O)c1 C(=O)(CCCCCS(N)(=O)=O)N1C(CNC(COC)=O)CCC(C)C1 C(C)(CCCC(=O)N1CCC(C(C)C#N)CC1)NC(c1cnc(SC)s1)=O c1(C(=O)NC2CC(C(=O)NC3CC3Cl)C2)ccncc1Cl C12(NC(CC(=C)C)=O)CCOCC1CN(C(=O)C(C)(C)CN1CCN(C)CC1)C2 c1(C(=O)NC2(C)CCN(C(=O)CNS(=O)(=O)C3CC3)C2)ccc2c(n1)COCC2 C(=O)(C(C(C)C)OC)N1CC(OC(C2CCN(C(=O)OC)C2)=O)C1 N1(C(CCCC(C)=O)=O)CC(CNC(=O)Cc2coc(C)n2)CC12CCC2 Cn1cc(C(N2CCN(C(=O)C(=CC3CCCCC3)F)CC2CF)=O)n(C)c1=O C1(CNC(c2ncsc2Br)=O)CC(O)CN1C(=O)CCc1nncs1 c1(C(N2CC=CC(C(N3CC(C)SCC3)=O)C2)=O)cccc2ccnn12 S(=O)(=O)(c1cc(C(=O)O)ccc1Br)NC(Cc1c(C)cc(C)cc1C)C(=O)O S(=O)(=O)(c1cnc(N2CCCC(F)(F)CC2)c(Cl)c1)NC(C)CO C1(C(=O)OCC)CCN(C(c2cnnn2C2CCOCC2)=O)CC1 C1(C(=O)NCc2c(C(N(c3ccn(CC)n3)C)=O)occ2)CC2CCC1CC2 c1(C(=O)NCC(CNC(=O)CC2CCC(=O)N2)OC)cc(OC)ccc1[N+](=O)[O-] C(=O)(C(F)C(CC)CC)N1C2CC(CNC(C=CCN(C)CC)=O)C1CC2 C(=O)(CS(=O)(=O)NC)N(C1CCN(C(c2cc(CN(C)C)c[nH]2)=O)C1)CC C1(C)(C(=O)NC(C)CCNC(c2scnc2C(F)(F)F)=O)CCS(=O)(=O)CC1 Cc1cc(C=CC(=O)NC2CC(O)C2CC(=O)NCC(N2CC=CC2)=O)on1 C1(NC(c2c(CC)c[nH]n2)=O)CCC2CC1CN2C(c1cccc(C#N)n1)=O N1(C(c2ccc(C)c(C)n2)=O)CCC2(CCCN2C(=O)C(C)C(C)(F)F)C1 C1(C2CCN(c3ncc4ccsc4n3)CC2)(NC(c2ccc3c(c2)CCC3)=O)CC1 C1(NC(C(F)=C(C)C)=O)CN(C(=O)CC(O)C(C)C)CC(C)(C)C1 C1(C2(C(=O)Nc3ccsn3)CC2)CCCCN1Cc1ncccn1 C12(C(=O)NCC3C(C)CCN3C(=O)CSS(C)(=O)=O)CCC(C)(CC1)OC2 N1(C(C(COC)N(C)C)=O)CC(N(C(=O)CSc2nncn2C)C)C(C)(C)C1 c1(SCC)ccccc1C(N1CC(CNC(c2coc(C(C)=O)c2)=O)CC1C)=O c1(OC)cc(CC(=O)NC2(C(=O)NCC3(N(C)C)CC3)CC2)c(F)cc1O C1(C(=O)NCC2C(CNC(CC(CC)(F)F)=O)C2)CC2COCC(C1)C2 C12(NCC(=O)NCC(C)C(F)F)CCCC1N(C(=O)OC(C)(C)C)CCC2 C1(N(C(c2nn(CC)cc2Cl)=O)CC)CCCN(C(=O)C(O)C2CCCC2)C1 c1(OC)ccc(C(N2CCC(CNC(c3ncccc3Cl)=O)CC2)=O)cc1F c1(NC2(SC)CC2)c[nH]c2ncnc(N3CCC(OCc4ccccc4)C3)c12 C1(C(N2CC(CC3CCC3)C2)=O)C=CCN1C(=O)CCCC1CCC1 C(=O)(C1=NOCC1)NCC1(NC(C(CC)OC)=O)CCOC1 N1(C(c2cccc(C)c2O)=O)CC=C(C(=O)NC2C3COCC23)CC1 C(=O)(C(C)(CO)NC(=O)CCc1cncs1)NCC(COC)OC c1(CC(=O)NCC(C2CC2)NC(C(CC=C)C)=O)coc2cc3c(cc12)CCC3 Cc1cc(Cl)c(C(=O)NC2CC2NC(C2CN3CCN2CC3)=O)cn1 c1(OC)cccc(NCCC(=O)NCCC2CCCN2C(=O)CNC=O)c1 C(c1ccccc1F)=CC(N1C(CN(C)C(C2CC3OC2C2CC32)=O)CCC1)=O N1(C(CCOC)=O)CCCC1(C)C(N1CCC(C(C)O)CC1)=O C=CCCC(CO)NC(=O)C(=O)NCCOCCN(C)CCOC N1(C(C2(F)C(C)C2)=O)CCC(F)(CNC(c2cc(C3CC3)ncn2)=O)C1 C1(C(N2CCC(NC(C(=O)OCC)=O)C(F)(F)C2)=O)CCc2cnc(C)n2C1 C(C1CN(C(=O)CSS(C)(=O)=O)Cc2ccccc21)NC(C1(C#N)CCCC1)=O C1(F)(CCNC(=O)CCC2CC(NC(=O)C(C3CC3)C3CC3)C2)CCCC1 c1(C(=O)NC2CC3(C2)CC(NC(C2CC2C2CCC2)=O)C3)nnn2c1CSCC2 C1(NC(=O)CN2CCCS2(=O)=O)CCN(C(c2ccnnc2O)=O)CC1O C(=O)(CC(C)C(F)(F)F)NCC(CC(C)C)NC(c1cn2c(n1)CCC2)=O CCC(C)C(C)N(C(=O)C(N)C1CNC1)C c1(CC)c(C(=O)NC2COCC2NC(C2CCS(=O)CC2)=O)cnn1C(C)(C)C CCC(CC(=O)NC(CNC(c1cnc(O)s1)=O)CC(F)(F)F)C(F)F C1(C(=O)NCCCCN(C(CC(=O)N(C)C)=O)C)CC2(CCOCC2)C1 N1(C(CNC(CN(C)C)=O)=O)CCOC(C)(CNC(=O)C(F)C2CCC2)C1 c1(NC(C(CC)NC(N)=O)=O)cccc(CN(C(=O)C(C)OC)C)c1.C1(SCC)CC1 N1(C(c2ccc(OC)cc2)=O)CCC(NC(=O)Cn2cccn2)C(C(C)C)C1 c1(C(=O)NC(CC=C)CNC(c2cncn2C)=O)ccc(C(C)C)nc1 C1(C)(C(=O)NCC#CC(=O)N(C(c2ccccc2)C)CC)C(C)(C)C1(C)C CCCCC(C)C(=O)N(CCN(C(c1cc(C(C)C)cnc1O)=O)CC)CC C1(CN(C(=O)CCNC(N)=O)C)CCN(C(c2cnc(C(C)(C)CF)o2)=O)CC1 C12(C(=O)NC3CCN(C(c4[nH]cc(C)c(=O)c4)=O)C3)CCOC1CCOC2 C=CCN=C(NCC1CCCN(C)C1)NCC1CN(S(=O)(=O)CC)C1 c1(OC)cc(C(=O)OCC2CC2)c(C(=O)Nc2nnc(SC)n2C)cc1OC C1(NC(COC)=O)CCC12CN(C(=O)C(c1cc(Cl)cc(Cl)c1)=O)C2 c1(OC)cc(CC(N2CC=CC(NC(C3CC(=O)OC3(C)C)=O)C2)=O)ccc1O C1(NC(CC2(COC)CC2)=O)CN(C(=O)Cc2ccn(C(F)F)n2)CC1(C)C c1(CCC(=O)N(CCNC(C=C2CCC(C)C2)=O)C2CC2)n[nH]c2ccccc12 C(CCCC(=O)N1CCC=CC1C(=O)NC1CCOC1)OCC c1(C(C(=O)NC(C2CN(C(=O)C3=COCC3)C2)C)C)cccc(Cl)c1 CCC(C)C(C)C(=O)N1CCC12CN(C(=O)Cc1ccccc1F)C2 Cc1ccnc(CNC(=O)C(c2ccoc2)NC(C2CCS(=O)(=O)C2)=O)c1 C1(CNC(CC=C=C)=O)(CO)CCN(C(=O)Cc2[nH]cnc2C)CC1 CC1=C(C(=O)N2CC(NC(c3cccc(C(F)F)c3F)=O)C2)CCCC1 N(C1CCOc2c(C)cc(C)cc21)C(CS(=O)(=O)NC)=O N1(C(C(C)OCC2CC2)=O)CCN(C)C(C(=O)NCC2CCOCC2)C1 c1(C(=O)NC(CN(C(=O)CCC2CCCOC2)C)(C)C)cncc(Br)c1 c1(C(=O)NCC(CC)NC(=O)CCn2ccc(=N)[nH]2)ccccc1F C1(NC(CCCOC)=O)CCN(C(=O)CCC(C)(C)N2CCOCC2)C(C)C1 c1(C(=O)NC2CC(C)OC2)cncc(CNC(C2CC2Cc2ccccc2)=O)c1 C1(C2CC2)(CNC(=O)Cn2cncn2)CCN(C(c2cccc(Cl)c2)=O)C1 C(=O)(CC1CCc2ccccc21)NCC1(OC)CN(C(=O)CCn2cnnn2)C1 N1(C(C2C=CC(=O)N=N2)=O)CC2(CCN(Cc3ccc(Cl)c(F)c3)CC2)C1 c1(OC)ccc(NC(c2nnnn2C(C)(C)C)c2ncco2)cc1C(F)F C1(NC(CCC)=O)CCC(C)(CNC(=O)C(C)C(F)(F)F)CC1 C1(NC(C(COC(C)=O)C)=O)CCN(C(c2cnc(C(F)(F)F)nc2)=O)C(C)C1 c1(C(=O)NCC2CN(C(c3c(OC)cc(O)nc3)=O)C2)c(Cl)sc(C)c1C C(=O)(C(O)C(C)(C)CC)NCC1(OCC)CN(C(c2cnc3sc(C)cn23)=O)C1 c1(C(C)NC(C2C3CCCC23)=O)cc(OC)ccc1OC(F)F C#CC(CNC(C1CCCN(C(=O)C(C)N2CC(C)C2)C1C)=O)C(C)C CC1CN(C(=O)Cc2nccn2C)CCC1NC(C1CCC2CC2CC1)=O c1(C(=O)NC(C(C)NC(=O)C=C2CCN(C)C2)(C)C)cc2nn[nH]c2cc1F C1(C(N(CCN(C)Cc2ccc(C)cc2Br)C)=O)CCc2ncnc(C)c2C1 C1(CNC(c2c(C)n(C(C)(C)C)nc2)=O)N(C(=O)C=CC2CC2)CCCC1(C)C c1(OC)ccc(C)c(C(=O)N(CC(O)CNC(c2cc3n(n2)CCO3)=O)C)n1 C1(CNC(c2cnccn2)=O)CC2(C1)CN(C(c1nc(Cl)sc1Cl)=O)C2 C1(C(CO)NC(C2(C)C(C)C2)=O)CCN(C(c2cccn2C2CC2)=O)CC1 C(CCSC)(CN=c1cc[nH]cc1S(=O)(=O)NCCCOCCOC)OC c1(C(=O)NC(CNC(C2CC2(F)F)=O)C2CCC2)cc2c(F)c(Br)ccc2[nH]1 C1(NC(c2scc(C)c2C)=O)CC2CC(NC(C3CCSCC3)=O)C2C1 Cc1nn2cc(C(=O)NCCC3CC(F)(F)CN3C(=O)C(C)CC(C)C)nc2s1 Cc1cc([N+](=O)[O-])ncc1C(=O)NC1CCC1NC(=O)CC1CCSCC1 CC(C)(C)CCCC(=O)N1CCC(C(=O)NCCC[Si](C)(C)C)C12CCC2 CCCCC(CNC(=O)C(C)(O)C1CCC1)NC(c1coc(Cl)c1)=O C=CCCN=C(NCc1ccc(Cl)nc1)NCc1cccc(Cl)c1 C1(C(=O)NCC2(O)CCOC2)CC12CC(NC(C1(CO)CCOC1)=O)C2 CC(C)C(C(=O)OC)NC(=O)CC1CCCN(C(c2cccnn2)=O)C1 C1(NC(C(Cc2ccoc2)NC(C2N(C=O)CCC2)=O)=O)CCCC(O)C1O c1(N2CCCC(COC)C2)nc(N2CCC(S(C)(=O)=O)C2)c2ncn(C)c2n1 N1(C(C(CC=C)(C)CC)=O)CCC(NC(c2sc(F)cc2C)=O)C2(CCC2)C1 C(=O)(C(C)CCCC(C)C)NC1C(C(=O)NCC2N(CC)CCC2)C1(C)C C1(NC(C(CC)OC)=O)CN(C(c2cccc(COC)c2)=O)CC1C c1(CN2CCC(C(=O)Nc3nc4sccc4[nH]3)C2)cc(Br)cc(Br)c1O c1(C(N2CC(O)(CNC(C3CCC(OC)C3)=O)C2)=O)ccc(SC(C)C)cc1 c1(CC(N2CC=CC(NC(=O)COC3CCCC3)C2)=O)ccc2c(c1)OCCO2 C(CCC(=O)NCC12CC(NC(C3CN(S(=O)(=O)C(F)F)C3)=O)(C1)C2)OCCC N1(C(CC2(C=C)CC2)=O)CC2(CC(NC(c3cc(OC4CC4)no3)=O)C2)C1 c1(C(N2CCCC(NC(c3c(C)ncnc3)=O)CC2)=O)cnn2c1OCC(O)C2 C(=O)(C(C)(C)CC(C)C)N1CC(C(=O)O)C(C)(C)C1.C(CC=O)=C(C)C c1(SCC(=O)NCC(=O)NCC2C(C(N)=O)COC2)cccc(C(F)(F)F)c1 c1(CC(=O)NCC=CCC(=O)NCC(C2CC2)OC)ccncc1C CC1CCCN(C(c2cc(=N)[nH]n2C)=O)C1CNC(c1ccc(CO)nc1)=O CCCCCCC(C)CC(=O)NCC(C)CCCNC(c1ccc(=O)n(C)n1)=O N1(C(C2(C(C)(C)OC)CC2)=O)CC2CCN(C(c3occ4c3CCOC4)=O)C2C1 N1(C(C=CCC)=O)CC(OC)C(CNC(C2CCCOC2c2cc[nH]n2)=O)C1 c1(CC(=O)N(CC(CNC(CNS(CC)(=O)=O)=O)O)C)c[nH]c2cc(Cl)ccc12 C12(CNC(C3=CC(C)CC3)=O)CCCC1CN(C(=O)CCCN1CCCC1)C2 C(=O)(CS(=O)(=O)CC)NCC(C)N(C(=O)C=Cc1cncn1C)CC c1(C(=O)NCCNC(COCC#C)=O)ccc2occc2c1 N1(C(CSCCOC)=O)CCC(CN(C(=O)CCC(=O)c2cnn(C)c2)C)CC1 CC#CCCCC(=O)N1CC(O)(CCNC(=O)CC2CCOCC2(C)C)C1 C1(NC(C(C)(C)SC)=O)CCCCCN(C(C2COCCO2)=O)C1 c1(C(c2nnnn2C2CC2)NC(C(F)(F)F)CI)cc(F)ccc1OCCO N1(CC(=O)NCC2(NC(CC=CCC)=O)CC(OC)C2)C(=O)CCCC1=O CCC(C(N)=O)OC.c12ccc(o1)C1CCCN1C2=O C1(CN(C(CCN(CCC)C)=O)C)CCCN(C(=O)Cc2ccn(C)n2)C1 CCCC(CCCNC(c1sccc1CN(C)C)=O)NC(C1CNC(=O)N1)=O C1(NC(c2cc(CC)n(C)n2)=O)CC2CC(C1)N(C(=O)CNC=O)C2 Cc1cn(C)nc1CNC(C1(CNC(=O)C=CC(=O)N(C)C)CC1)=O c1(C(=O)NC(CSC)CNC(=O)CC(O)C2CCCC2)cnc(O)cc1C c1(N(C(C(c2cccc(C)c2)=O)=O)C2CCNC2)ccn2ncc(Br)c2n1 C(=O)(CCCCCSC)NCC(C(=O)NC(c1ccncc1)C)OC N1(C(c2sccc2Br)C(=O)NCCSC)CCCC2(CC1)CCN(C)CC2 C(=O)(C(CCC1CC1)SC)NCC(CC)NC(=O)Cn1cc(C(C)O)nn1 N1(C(c2cc(C)nn2C)=O)CC2CCCC1(CNC(=O)CC1C=CS(=O)(=O)C1)C2 C1(C(=O)OC)CNC(=O)CN1C(=O)OC(C)(C)C.c12ccc(c(C)c1)[nH]2 c1(OC)cc(C(N2CCC(NC(c3ccc(Cl)[nH]3)=O)C2)=O)ccc1Cl C1(NC(C(CCC)NC(C)=O)=O)CN(C(c2ccc(OC)o2)=O)CCC1C N1(C(C(C)OCCN(C)C)=O)CCCC(CO)(NC(C2CC2C2CCC2)=O)C1 c1(NC(=O)NCC=CCO)ccccc1SCc1ccccc1.C1(N)COC1 c1(CCC(=O)NC2C(NC(C3(C)N(C)CCC3)=O)COC2)cc2ccccc2[nH]1 N1(C(C2CCCN2C(C2CCCC2)=O)=O)CC2(CCC2)C12CCC2 c1(CCC(CO)N(C)Cc2cc(Cl)n(C)n2)ccccc1F c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)cc(-c2ccncc2)[nH]n1 Cc1ncc2n1CCC(C(=O)NC(C)CNC(=O)C=Cc1ccnn1C)C2 C1(C)(C(=O)NCCOCC)CC(O)CN1C(C1COCC(C)O1)=O N1(C(c2n(C=C)nnc2)=O)CC(C(=O)NC2CSC2)CC12CCC2 N(C1CC2(CCCC2)c2ccccc21)C(N1CCCC1CCc1cccnc1)=O C(CCCCC(=O)N1CCCC1CN(C(=O)CC1C(=O)NCCC1C)C)=CC c1(-c2nnc(N(C(C#C)C)C)n2CC(C)C)ccc(C#N)cc1 C(CCF)(C(=O)NCCC1(O)CCCC1)NC(c1c(C)c[nH]n1)=O c1(-c2c(C(=O)NOCCc3ccccc3)cc(C)s2)c[nH]c2ccc(OC)cc12 c1(C(N2CC(C)(CNC(=O)CC3CCCCC3)OCC2)=O)ccn2c1CCCC2 Cn1cc2c(C(=O)NCC3COC(CN=c4[nH]cnc(Cl)c4F)C3)cccc2n1 N1(C(Cn2c(C)nnn2)=O)CCC2(CC1)OCCC2NC(c1ncccc1Cl)=O c1(N2CCC(CSC)CC2)nc(N2CCC3CCC(C2)N3C)c2ncccc2n1 c1(NC(CN(C(c2nc(CC)sc2)=O)C(C)C)=O)cnc2ccnn2c1 Cc1c(C(=O)NCCOCCNC(C2CCOC(=O)N2)=O)[nH]ccc1=O c1(CC(N2C(C)(C)C(NC(=O)C=CCN(C)C)CC2)=O)ccc2c(c1)CCCS2 N1(CC(=O)NCC23C(CN(C(C(C)CC4CC4)=O)C2)C3)CCc2ccccc21 N1(C(CCc2scc(C)c2)=O)CCN(C(C2CCOC2)=O)CC(O)C1 c1(NC(C(C)(C)O)=O)cccc(C(N2CCCC(Nc3ncccn3)C2)=O)c1 CC1CCN(C(=O)C2=COCC2)C1CNC(c1cc(-c2ccco2)[nH]n1)=O CC1CCCCC1(CNC(c1cc2n(c1)CCC2)=O)NC(c1cnncc1O)=O c1(OC)ccccc1CN1CCC(C(=O)C(F)(F)Oc2occc2OC)CC1 CCC(CC(=O)N(C)Cc1ccc(C)cn1)N(C(=O)Cc1ccc[nH]1)C CCCC(C#N)C(=O)N1CC(CCO)(NC(c2c(C)csc2C)=O)C1 CCC(F)(F)CC(=O)NCC(C)CN(C)C(c1ccc(OCCF)cn1)=O c1(OCC(=O)N(C2CCN(C(CC3(C(=C)F)CCC3)=O)C2)C)ccc(C)c(C)c1 CC(CC(=O)N1CC2(NC(=O)CN(C)S(N)(=O)=O)CCCC2(F)C1)CC(F)(F)F c1(C(N2CC(NC(CC(CCC)(C)O)=O)C(C)C2)=O)c(O)cnc2ccccc12 c1(Sc2ccccc2)nn(C)c(CN(C2CCN(c3ccncn3)C2)C(C)=O)c1Cl c1(CN2CC(n3cc(CNC(c4cc(CC)c(C)s4)=O)nn3)C2)cc(F)cnc1Cl O(NC(=O)CCCCCNC(c1cccn2nccc12)=O)CC(C)O C(C(C(=O)N1CCC(C)(F)CC1)C(C)C)NC(CC(CC)C1CCC1)=O c1(C(N(C2CCC(NC(C=CCC)=O)CC2)C)=O)ncc(F)cc1F c1(C(=O)NC(C)CCNC(=O)CN2C(=O)CCC2=O)nnn2c1CCC2 N1(C(C(C(C)C)CO)=O)CCN(C(c2ccccc2F)=O)C(c2cncnc2)C1 C1(CCn2cc(-c3cnc(OC)c(C)c3)nn2)CC(F)(F)CN1C(C1CC1Cl)=O c1(-c2cccc(N(C(C3CCCC3)=O)CC)n2)ccc2ccccc2c1 N1(C(C(C)Cc2cccs2)=O)CCCC2(C1)CN(C(c1cn(C)ccc1=O)=O)C2 c1(C(=O)NC2C(CNC(CCC=C)=O)COC2)ccc2c(c1)nc(C)n2C1CC1 C(C1=CCN(C(C2CC3CC3C2)=O)CC1)NC(C1(COC(C)C)CC1)=O c1(CCC)sc(N2CC3CC2(C(=O)OC)C3)nc1-c1cnccn1 C(=O)(CCCC(=O)N(C)C)NC(CNC(C(C)Nc1scc(C)n1)=O)(C)C(C)C C12CCN(C1)C(=O)C(C)(C)NC2=O.C(CC(=O)Nc1ccco1)OCCC N1(C(C2C=CCC2)=O)CCC2(CC1)CCN(C(C1(c3ccc(F)cn3)CC1)=O)C2 C(=O)(C(C)(C(C)C)OC)N(CCC)Cc1cc(C)sc1C N1(C(NS(NC)(=O)=O)c2nnnn2C)CCOCC1c1ncn(C(C)(C)C)n1 Cc1cc(Cl)cc(N)c1C(N1CC2CC2(CNC(c2cc(C(N)=O)no2)=O)C1)=O CC1CC(C(=O)N(CC(=O)NCCC(O)C(F)F)C2CC2)CN1C c1(SCC)cccc(C(=O)NCC23CC2CN(C(c2ccnn2COC)=O)C3)c1 CCCC(C(=O)NC(C)(C)C(=O)NC(C)(C)C(O)CO)N(C)C Cc1ccc(F)c(C(=O)NC(C(=O)NC(CO)CCCO)C(C)C)n1 C1(CC(=O)N(CCO)CC)CN(C(=O)C(C)c2cc[nH]n2)C(C)(C)C1 C(C(CNC(=O)C=Cc1ccco1)C(F)(F)F)NC(COC(CC)C)=O n1(CC)nc(C)c(CC(=O)N(CCCNC(c2c[nH]c(=N)s2)=O)CC)c1C C1(N(C(c2cc(C(C)NC(=O)Cc3ccccn3)no2)=O)C)CCOC(C)C1 C1(C(c2ccccc2)N(C)Cc2nc(C)sc2)CC(=O)CC(=O)N1 Cn1nc(-c2nnc(CN3CCCC(C4CCCCO4)C3)o2)ccc1=O N1(C(CCC(C)C)=O)CC2CC(NC(C3(c4ccc(Cl)nc4)CC3)=O)CC2C1 c1(C(=O)NCCC(C)NC(COc2c(C)cccc2C)=O)ccc(C)n(C)c1=O N1(C(CC2CC(=C)C2)=O)CC2CCC(NC(c3cncc(COC)c3)=O)CC2C1 C1(CNC(CCc2cn(C)nn2)=O)CN(C(=O)CCSCC(F)(F)F)C(C)(C)C1 CS(=O)(=O)c1cccnc1C(=O)NCC1CN(C(=O)C2CC2)CCC1C(F)(F)F c1(C(=O)NCCOCCCN(C(CC)=O)C)ccsc1CC C(=O)(C(C)C(F)(F)F)Nc1sc(C(=O)NCC(CCCC)NC(=O)OC)c(C)c1 N1(C(C(C(C)C)NC(c2cn(CC=C)nc2)=O)=O)CC(O)CC1(C)C C(C(C)NC(c1n[nH]cc1C)=O)(C(C)C)NC(C=CCC)=O C(=O)(CC(C(F)F)N1CCOCC1)NCC1(C)CC(NC(=O)CC2(O)CCC2)C1 C1(C(C)=O)CCN(CC(=O)OC)C(C)C1.n1(CCC(=O)NCC(C)C)nc(C)nc1C C1(CC)CNC(=O)CN1C(C1(CC)CCN(C(C2CC(OCC)C2)=O)C1)=O Cc1cc(C(=O)N(C2CC(NC(C3(SC4CC4)CC3)=O)C2)C)c(C)n1C(C)C C1(NC(CCc2cncc(C)c2)=O)CCN(C(=O)Cc2ccsc2)C(C)C1 C#CCCCCCCC(=O)NCC12CCC1CN(C(c1ccc(CO)cc1)=O)C2 N1(C(CN2CCN(C(c3nncc(OC)c3)=O)CC2)=O)CCCC2(C1)N=N2 N1(C(CSCCC#N)=O)C(C(=O)NC2(C(=O)NCCO)CCC2)CC2CC12 CC1CCC(CC(=O)NCCNC(C2(c3cc[nH]n3)CC2)=O)O1 c1(C(N2CCC(O)(CNC(C3(C=C)CC3)=O)C2)=O)cc(F)cc(Br)c1F N1(C(COC(CC)CC)=O)CCCC(C2CN(C(C(C)CC)=O)C2)C1 C1(C(=O)O)CC(=O)NC1.C12(C(N(CCO)CC)=O)CCC(C(C)C)(CC1)C2 C(CNC(=O)CC1=CCCC1)(C(C)C(C)C)NC(C=C(COC)C)=O c1(C(=O)NC(CC2CN(C(c3cnc(C)o3)=O)C2)C)cc2ccc(Cl)cn2c1 C1(N(C)C)(CC)CCN(C(=O)CC(COC)NC(=O)Cn2cccnc2=O)C1 N1(C(C(CC(C)(C)NC(c2cccc(CO)n2)=O)F)=O)CCC2(CCCO2)CC1 c1(C(N(C)CC2CN(C(CCOCC)=O)C2)=O)cc2ccc(OC)nc2[nH]1 c1(C(=O)NCC2(OC)CN(C(C3CN(C)CCO3)=O)C2)cnc(C)nc1O C1(C(N2CC(=C(CNC(c3c(CC)cno3)=O)F)C2)=O)CC1C1CCCC1 c1(OC)cc(C(=O)NC2CCCCN(C(=O)C(F)C3CCC3)C2)cc(C)n1 N1(C(=O)NC2C(C(=O)O)CC(F)(F)C2)C2CCCC1CC1(CCC1)C2 C1(N(C(=O)Cn2cc(C3CCC3)nn2)C)CC2CCC(C1)N2C(=O)C(F)F C1(C(=O)NCC2(O)CCN(C(c3c(C)sc(O)n3)=O)C2)CN2CCCC1C2 C(CO)(C(=O)NCC1(NC(=O)CCOCC(F)F)CCCC1)OC C1(CCC)(C(=O)N(C)CC2(CNC(=O)C(C)(C)N3CCCC3)CC2)CCNC1=O CCCCCC(=O)N1CCCC(CCCCNC(C2(COC)CCCO2)=O)C1 C1(NC(C2N(C=O)CCC2)=O)CCCN(C(c2ccc(Cl)cn2)=O)CC1 Cc1ccc2c(C(=O)NCC3CCCCN3C(=O)C(F)F)coc2c1 C(=O)(CC1=CCOCC1)NCC(CNC(C(N1CCCCC1=O)C)=O)CO CC1CN(C(=O)Nc2nc(-c3ccccc3)cs2)CCN1CC(F)F C(CCCCC(=O)N1CC(F)(CNC(c2cc(CC(C)C)[nH]n2)=O)C1)OC c1(CC(=O)NC)csc(N(c2ccccc2)C(=O)Nc2nc(C(F)F)cs2)n1 Cc1nn(C)c2sc(C(=O)NC(C)CNC(=O)CC3CC4(CCCC4)CO3)cc12 C1(CC(=O)N(CCC(=O)NCCc2c(C)n[nH]c2)CCO)CCC(C)CC1 CC1CN(C(C2CC(F)C(=O)N2)=O)CCC1CNC(=O)CN1CCN(C)CC1 CCCCCC(C)(C)C(=O)NC(CNC(=O)C(C)(C)OC)C(C)C c1(C(=O)NC(C)CC(C)NC(=O)C(C)(F)F)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 c1(NC2(CNC(C(C)N3CCC3)=O)CCCCC2C)ncnc2sccc12 N1(C(c2ccc(SC)o2)=O)CC2(CCC(Nc3nnccc3C(F)(F)F)C2)C1 c1(C(=O)NCC2N(C(CNC(C)=O)=O)CCC2C)c(C)cc(Cl)cc1C N1(C(Cc2cccc(CS(C)(=O)=O)c2)=O)CCN(C(C2CCC2)=O)C(C2CC2)C1 Cc1ccc(NC(=O)C(N2CCOCC2(C)C(F)F)=O)cc1Br CCCC(C#N)C(=O)NCC1(O)CCN(C(=O)CC2CCCC2(C)C)CC1 C=C1CC(C(F)(F)F)(C(=O)NCC(C)CNC(c2nncn2CC#C)=O)C1 c1(OC)ccc(C(F)(F)F)cc1C(=O)NC1(CNC(C2COCC(C)O2)=O)CC1 CC(C)CC(O)CC(=O)N1CC(NC(c2ccc(C(F)F)o2)=O)C2(CCC2)C1 N1(C(CS(=O)(=O)N(C)C)=O)CCCC(C)(CNC(C23CC=CC(C2)OC3)=O)C1 C1(CNC(C2(COCC)CC2)=O)CN(C(=O)CC(C)(C)C)CC1O CC1(C)CCOC(C(N2CCC(NC(=O)CCCn3ccnn3)C(O)C2)=O)C1 CC#CC1CCN(C(C2CCCC2CNC(=O)NC2(C)C=CCCC2)=O)C1 C1(NC(C(C2(C)CCCC2)C)=O)CC(CNC(C2(C)CCSCC2)=O)CC1O C(C(C(=O)OCCc1nc(OC)ns1)N(C)C)OC C=CCN(OC)C(=O)C1CCC2(CC2)N1C(C1CCCN1CCC)=O c1(C(N2C3CC(CC(NC(C)=O)C3)C2)=O)ccc2nc(S)[nH]c2c1 Cc1cccc(CNC(C2CC(F)CN2Cc2cnc(C(C)(C)C)nc2)=O)n1 C(=O)(C(CNC)C(C)C)NC1CC(CC)OCC1 c1(C2(C(N3CC(OC)C(NC(C4CC4(F)F)=O)C3)=O)CC2)c(F)cccc1Cl C(=O)(C(C)CCCC(C)C)N1CCCC(CCNC(c2n(C=C)ncc2)=O)C1 O=C(C1OCCc2c(F)cccc21)NC1(c2ccc(F)nc2)CC1 CCCCC(C(=O)NCCN(C)C(C1(c2ccccc2C)CC1)=O)N(C)C N1(C(c2cnn(C)c2N)=O)CCN(C(C2CCOC2)=O)C(C2CCC2)C1 C1(CC(=O)NC(CCC)C)CCN(C(=O)COCCCN(C)C)CC1(C)C N1(C(c2c(CC)ccc(F)c2)=O)CCC2CCN(C(c3ccc[nH]3)=O)C2C1 Cc1c(C(=O)NCC2(CNC(c3ccc(Cl)o3)=O)CCC2)cnn1CCO CC(CCCNC(=O)CCCc1nccs1)NC(=O)CCc1cscn1 C1(NC(c2c(F)ccc(C(C)C)c2)=O)CCN(C(=O)CCC(F)(F)F)CC(O)C1 N1(C(C=CC)=O)CCC2(CCC2)C(CNC(=O)CCC(CC)OC)C1 c1(C(N(C(CCNC(C2CC(O)(CC#C)C2)=O)=O)CC=C)C)cc(C)cnc1F C1(c2nnc3n2CCN3C)CCCC2(C1)CC2(F)F.CC1CSC(C(F)(F)F)C1 C12(NC(CCc3cc(C)nc(C)c3)=O)CCC(CN(C(C3(Cl)CC3(C)C)=O)C1)C2 c1(C(N2CC(O)(C(C)NC(C3CC(CF)C3)=O)C2)=O)ccnc(O)c1Br C1(C(=O)NC2CC(CNC(c3cc(O)ncn3)=O)C2)CCCC2(C1)CC2(F)F Cc1nn(C)c2ncc(C(=O)NCC3CCC3NC(=O)CC3CC34CC4)cc12 c1(C(=O)NCCN(CCC)C(C2CC2F)=O)sc([N+](=O)[O-])cc1Cl CC1CCCCN1CCC(=O)NC1CC(C)(CNC(=O)C=CBr)C1 Nc1cnc(NCc2ncon2)c(Cl)n1 C1(CNC(COCC)=O)CCC(N(C)C(C2(c3cc(C)on3)CC2)=O)CC1 N1(C(C2C(=C)CC2)=O)CCOCC1CCNC(=O)CC1CCN(S(C)(=O)=O)CC1 c1(C(N2C3C(NC(CN(C)CC)=O)C(CC3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] n1(CC)nc(CN2CCC(N3CCC(N)C3)CC2)c(C)n1 c1(Cn2c(C(=O)Nc3n(C)nc(Br)c3)ccn2)ccccc1C#N C(c1ccc(F)cc1)=CC(=O)NC1CCC(F)(CNC(c2ccc[n+]([O-])c2)=O)C1 c1(CC)ccoc1C(=O)NCC1(CCN)CC1.C1(C(=O)C2CC2)CC(CF)C1 C12(NC(c3c(O)ccc(OC)c3)=O)CCCCC1CN(C(=O)CN(C)C(C)C)C2 c1(N2CCOCC(NC(=O)NCc3ccc(C)cc3)C2)cc(C)c(C#N)c(C)n1 c1(C(N(CC(C)(C)CNC(c2ocnc2C(F)F)=O)CC)=O)cc(F)cc(F)c1 N1(C(Cc2cn(CC)nc2)=O)CCCC1(C)CNC(C1CC1F)=O C(C1COc2ccccc21)N1C(=O)N(C)C(c2cc(Br)ccc2C(F)(F)F)C1=O CC1CC(O)CCN(C(=O)C(Cn2ccnn2)NC(c2ccn(C)c(=O)c2)=O)C1 Cc1nc(C(=O)NC(c2ccc(F)cc2)CNC(C2(Br)CC2)=O)sc1C Nc1c(C(=O)NC2CC2CNC(C2(c3ccccc3)CCC2)=O)cnn1CCO Cc1cc(C)n(CCC(=O)N(C23CCC(CC2)C3)C)n1 C12(C(N(CCCNC(CC3CC(OC)C3)=O)C)=O)CCC(N=[N+]=[N-])C1C2 c1(OC)cc(C(=O)NCC2(CNC(=O)CCCSC)CCC2)ccc1Cl C12(C(N(C3CCN(C)C3)C)=O)CC1CCN2C(=O)CCCN(C)C1CC1 N1(CC(C)C)CCCC(C(=O)NCCCCNC(c2cncc(C3CC3)c2)=O)C1 C1(CC)CN(C(c2cnn(C)c2Cl)=O)CC1NC(c1sc(C)nc1C)=O CC1CN(C(=O)COc2ccon2)CCCC1NC(c1ccccc1Cl)=O CC1N(C(C2CC23CC(NC(=O)C#CC2CCOC2)C3)=O)CCOC1(C)C C(=O)(CC(CC)C(C)(C)C)N(CCC)CCNC(c1sc(C(F)(F)F)cc1C)=O CC1CCN(CC(N2CCCC2CN(C)C(c2cc(Br)cs2)=O)=O)C1 C1(C(=O)NCc2cccc(OCC3CCOC3)c2)CCn2c(cnc2Br)C1 CCCC(C(=O)NCC(C)(C1CC1)NC(=O)CCC(C)SC)S(N)(=O)=O c1(C(=O)NC2CC(C)N(C(c3ccc4occc4n3)=O)C2)ccc2c(c1)CCN2 c1(C(=O)NC(C(=O)NCC(CC)CC)C2CCCO2)ccc(C#N)c(C)n1 CC(CCCOC(C)(C)C)N(C)C.C(C(C)(C)O)N1C(=O)C1 C1(C(=O)NCc2ncc(C(F)(F)F)s2)CCN(S(=O)(=O)C(F)(F)F)CC1 CCC(CC)CN=c1cc(C)nc(N2CCCN3C(=O)CCC3C2)[nH]1 c1cccc(CO)c1.c1(CNC(CNC(C)=O)=O)nc(CNC(=O)C=C(C)C)cs1 N1(CC2CCC(C)O2)CC2CC(NC(c3cnn4c3CCC4)=O)CC1C2 C1(CC)(CO)CCN(c2ccnc(NCc3ccccc3OC(F)(F)F)n2)C1 c1(CC(=O)NCCC2(O)CN(C(COCCOCC)=O)C2)ccc2c(c1)CCC2 c1(CC(=O)NC2(CC)C(C(=O)NC3CC(CC)(CC)C3)CC2)cccnc1C CC1CCOC(C(=O)NC2CCCC(NC(=O)C3=CCOC3)C2)C1 c1(C(=O)NCCCNC(=O)Cn2cccn2)cnc(C2CC2)s1 C(C)(C)(CCCNC(C1CCCN1C(=O)C(C)(C)C)=O)OC C1(NC(C2CCCC(OC)C2)=O)CCC2CN(C(=O)COC(F)(F)F)CC2C1 c1(OC)cnc(C(=O)NC2CCN(C(c3ns[nH]c3=O)=O)C2C)cn1 N1(C(COCC)=O)CCC(CN2CCN(C(=O)C=Cc3cnc[nH]3)CC2)CC1 C1(C(=O)NCC(C)N(CC)CC)CN(C(=O)C=C2CC2)CC12CCC2 C(C)(C(=O)N1CC2CC2(CNC(C2CCCS2)=O)C1)(C(C)C)NC(C)=O c1(C(=O)NCCCCC)cc2cc(-c3cccc([N+](=O)[O-])c3)cnc2[nH]1 N1(C(C=C(COC)C)=O)CC(C)C(C)(C(=O)Nc2ccc(F)c(C)c2)C1 C1(NC(C(CNC(=O)COc2cccnc2)N(C)C)=O)COCCC1(F)F C=Cn1nncc1C(N1CCC(C(F)CNC(=O)CCSCCCC)CC1)=O c1(OC(CC)C(=O)N2CCC2CNC(=O)C=C(C)Cl)ccc(CCC(=O)OC)cc1 c1(C(N2CC(C)C(NC(=O)CC(F)(F)Cl)C2)=O)c[nH]c2c(F)cccc12 c1(C(N2CCC(CC(C)NC(C3CCC(O)C3)=O)CC2)=O)cccc(N)c1F N1(C(C(C)O)=O)CCCN(C(c2cc3n(c2)CCC3)=O)CC1 c1(-n2c(-c3ccnn3CC3CCOCC3)nc(CCOC)n2)cc(Cl)nc(Cl)c1 C1(NC(CCc2ccc(OC(C)C)cc2)=O)C2CCC1N(C(=O)C(O)C(C)C)C2 N1(C(C2CC(N(C)C)C2)=O)CCC2(CC1)CC2NC(c1ccno1)=O C1(C(=O)NCC2CC(NC(CN(C3CC3)CC)=O)C2)CC1C1CCCCC1 C(=O)(C(C#N)C(C)(C)C)NCC1CCN(C(CS(=O)(=O)NC)=O)CC1C c1(C(=O)NCC(CO)NC(=O)CCc2nc[nH]n2)ccc(C2CC2)s1 CC1CCCC(C)N1C(C1CCCN(CCOc2ccc(C(F)(F)F)cc2)C1)=O n1(CC(=O)NC(C(CO)NC(c2ccc(=NC)[nH]c2)=O)C)c(C)cc(O)cc1=O C1(C)(C(=O)OC)CCC1(C)C(=O)NC1CN(C(C2COCCO2)=O)C1 C#CCC(CC(F)F)NC(=O)C(CNC(c1cnncc1C)=O)CCC N1(C(C(CC)(F)F)=O)CCC2(CCC2)C(CNC(=O)C(CC)NC(N)=O)C1 c1(Sc2c(NC(C3(C)CC3(F)F)=O)cccc2)cc(F)cc(F)c1 C1(CN(C(CCC)=O)C2CC2)CCCN1C(=O)C(=O)NC C1(C)(n2cc(C3(C)CCN(C(C(CC)C(C)(F)F)=O)C3)nn2)CCCCC1C c1(-c2cn(CC(=O)NCC3(OC)CCCOC3)nn2)c(F)cncc1F C(=O)(C1=CCN(C(C2CCC(CO)CC2)=O)C1)NC(CCC)(C)CO N1(C(C(F)OC)=O)CCCC(N(C)C(c2coc(O)n2)=O)CC1 N1(C(CCc2n(C)cnn2)=O)CCN(C(c2[nH]ncc2C#N)=O)C(C2CCC2)C1 C(=O)(C(F)(F)CC(C)C)NCC1(C)CCC(NC(C(C)=CC)=O)CC1 C(C(=O)N1CCCC1C1CCN(C(=O)CCC(C)SC)C1)(C(C)C)n1ccc(C)c1 C1(O)(CN(C)C(c2ccnn2-c2ccncc2)=O)CCCN(C(=O)CC2CC2)C1 C(N=c1ccnc(C(C)(C)C)[nH]1)C1CC(OC)C1.C1(C(=O)N)(CCF)CC1 C1(NC(C(CCOC)C)=O)CC2CCC1CN(C(c1ccc(Br)cc1C)=O)C2 c1(C2(C(CCC)C)CCC2)nnc(N(c2ccccc2)C)n1CC1CCCC1 C1(NC(C(COC)(F)F)=O)CC2(C1)CC(C(=O)Nc1cccc(Cl)c1Br)C2 C1(C(=O)NCCCCCCNC(c2c(CC)nco2)=O)CCn2c(cnc2C)C1 c1(NCCCOC)ccc(C)c(N(C)Cc2ccc(C)nc2OC)c1 NS(=O)(=O)c1ccc(F)c(C(=O)NC2CCC(CNC(=O)C=CCF)C2)c1 CC(CNC1(c2ccco2)CC1)C(=O)N(C)CC1CCO1 C(c1ccoc1)=CC(=O)N(CC(CNC(CCOCC(C)C)=O)O)C C1(CC(=O)N(C2CCCC2C#N)C)CN(C(c2cncs2)=O)C(C)(C)C1 c1(CC(=O)Nc2ncc(C3CC3)s2)ccc(O)cn1 C1(CNC(C=Cc2ccc(C)s2)=O)CN(C(=O)CC2CC2C(F)(F)F)CCC1C c1(N2CCC(C)(C(=O)NC)C2)cccc(S(=O)(=O)NCc2cc(CO)ccn2)n1 C(=O)(C(F)(F)CCc1ccccc1)N1C(CNC(=O)CCCn2cccc2)CC1 c1(C(=O)NC2C(NC(Cc3cc(OC)no3)=O)CCC2)ccc2cnnn2c1 C1(CC(N2CCC(NC(C3(CSC)CCC3)=O)C2)=O)CC2(CC2)CO1 CC1CCCC(C)N(C(=O)CN(C)CCN(C)C)C1 c1(C(=O)NC(CCOC)CNC(=O)C=C(C)C)cc(N)cnc1Cl C#Cc1ccc(C(=O)NCCC(C)(C)COC)cc1Cl C1(C(=O)NCCOCCC=C)C(C)CN1C(=O)CCCSC N1(C(c2[nH]cc(C#N)c2)=O)C2CCC1CN(C(=O)CCn1cnnn1)C2 N1(C(c2cnc(CC)s2)=O)CC(N(C)C(c2cnc(C(C)(C)C)o2)=O)C(C)(C)C1 C1(NC(=O)C=Cc2cccnc2)CS(=O)(=O)CC1NC(c1cc(C(F)F)cs1)=O C1(c2cn(C(C)C)nn2)N(C(c2cc3n(c2)CCCC3)=O)CC12CCOCC2 c1(C(N2CCC(CCNC(C(C)C(C)(F)F)=O)C2)=O)ccc2c(c1)NC(=O)C2 CC(CCC(F)(F)F)(C(F)(F)F)NC(C1CC(NCc2ccccn2)C1)=O C1(C(=O)NC2CCCC(O)CC2)(CC)CCN(C(=O)C(CC2CC2)OC)CC1 C1(NC(Cn2ccc(C)n2)=O)CC(C)CN(C(=O)CCCN(C)C)C1 C1(CC)C2=CC=CC=CN(CCCCNC(C)C)C(=O)C2(C)NC1=O Cc1cc(C)n(C(C)C(N2CC3C(CNC(C4CC(C5CC5)C4)=O)C3C2)=O)n1 c1(CC(=O)NCC2C(NC(C3CCC(C)O3)=O)COC2)cc(F)c(F)cc1F C1(CC(=O)NC(CC=C)CC)CN(C(=O)CCn2ccnc2C)CCC1(C)C Cc1cc(C)n(C(C)C(=O)NC(CO)C(C)NC(=O)CNc2nccs2)n1 N1(C(C2C(C=C)OCCC2)=O)CC(F)(F)CC1(C)CNC(=O)CC C1(NC(C(C)NC(N)=O)=O)CCN(C(C23CCC(C#N)(CC2)CC3)=O)CC1(C)C C1(CNC(c2nnnn2CCCC2CC2)CCC)CC12CCC(F)(F)CC2 c1(C(N2CCC(CN(C(=O)C3=NNC(=O)C3)C)C2)=O)ccc2oc(O)nc2c1 c1(C(=O)NCCC(C)NC(c2nc(C)n(C)n2)=O)cc2ccc(F)cc2cn1 C1(NC(C2(NCC(=O)Nc3c(N(C)C)nccc3)CC2)=O)CCC(C)(C)CC1 Cc1scc(C(=O)Nc2cccc(NC(=O)C=CS(C)=O)c2)c1Br c12cnc(nc1)s2.c1(OC)nc(-c2ccccc2C(F)(F)F)sc1C C(=O)(C1=C(F)CN(C(C2CC23CCCC3)=O)CC1)NC(c1cccs1)(C)C c1(CC(=O)NC2CCN(C(COCC#C)=O)C2C(C)(C)C)c[nH]c2cccnc12 N1(C(Cn2ncn(C)c2=O)=O)CC(F)(F)CC1C(=O)Nc1ncc(F)cc1F C1(C(N2C(CN(C(=O)CCSC)CC)CCC2)=O)CCC2CC(C)CN2C1 C(CCCCC(=O)NC1CCCCC1N(C)C(c1cc(C(=O)OC)co1)=O)=CC c1(C(=O)NC2CC(NC(C(C=C)O)=O)C2)nsc2c(OC)cccc12 C(CN=c1nc(S(C)(=O)=O)cc[nH]1)C1CCN(C(C2=NOC(C)C2)=O)C1 C1(C(=O)C(F)(F)F)(NC2CC(CC)C2)CCOCC1 O=C(C1CCCn2cnnc21)N1CC(C2(NC(C3CC(C(F)(F)F)=NO3)=O)CC2)C1 C1(NC(CC(c2ccc(C)cc2)C)=O)COCCN(C(=O)C=C(Cl)Cl)C1 CC1CCOC1C(=O)NC(C1(O)CN(C(c2c[nH]c(=N)o2)=O)C1)C C(C(C)(C(C)C)NC(=O)CCn1ccnc1)NC(C(n1ncc(C)c1)C)=O c1(OC)ncc(C(=O)NC2CC(CNC(C3CCSCC3)=O)C(O)C2)cn1 C1(CC(=O)NCCC(CNC(COC(CC)(C)C)=O)O)CCC(C)(C)O1 N1(C(C2(n3cc(C)cn3)CC2)=O)C2CCCC1CN(C(c1ccsc1CC)=O)C2 N1(Cc2cc(C)[nH]c2C)CC2(CCC(NC(C34CC(C(F)(F)F)(C3)C4)=O)CC2)C1 c1(OCC(N2CC(CNC(C3C4CNC(=O)C34)=O)C2)=O)cc(Cl)cc(Br)c1 c1(C(=O)NCC(C)NC(CN(C)CC)=O)ccc(S(=O)(=O)N(C)CC)o1 c1(C(=O)NCC2CN(C(Cc3c(C)cco3)=O)C3C2C3)cccc2ncnn12 C1(C)(C(=O)NCC(NOCC(CC)C)=O)CC(=O)N(C)C1 Cc1cc(CN2CCN(S(=O)(=O)CC3CNC(=O)CO3)CC2C)ccc1O N1(C(c2ccc3[nH]c(=N)sc3c2)=O)CC2ON=C(CNC(C3(Cl)CC3)=O)C2C1 Cc1ccc(CC(=O)NCCC(C)NC(c2ccc(=O)n(C)n2)=O)cc1Cl Cc1cnn(CCC(=O)NCC2(CNC(=O)CCOC3COC3)CCC2)c1 C(CCCC(C)NC(=O)CS(N)(=O)=O)NC(Cc1nc(C)oc1)=O C1(CNC(C(F)=C(C)C)=O)CN(C(=O)CCc2cnn(C)c2)CC(C)(C)O1 C1(C(=O)NC(CC)CO)Cc2nccnc2CN1C(=O)C1=NN(C)C(=O)CC1 CC1=CC(F)(C(=O)NCC2CCN(C(=O)CCc3nc[nH]n3)C2(C)C)C(F)=C1 Cc1cc([N+](=O)[O-])nn1CC(=O)NCC12CC(CN1C(=O)C=Cc1cc[nH]c1)C2 Cc1ccn(CC(=O)NC2CCC(C)N(C(c3scc(C)c3C)=O)C2)c(=O)c1 N1(C(C(CCOC)C)=O)CC2CCCN(C(C34CCCC3C4(F)F)=O)C2C1 c1(C(=O)NC2CN(C(C(C3CC3)SC)=O)CC2C)c(F)c(F)c(F)c(F)c1F Cc1ccc2scc(C(N3CCC(CNC(=O)C(F)C(F)(F)F)C3(C)C)=O)c2c1 C(C)(CN=c1cc(Nc2cc3c(nn2)CCC3)nc(C)[nH]1)N(CC)CC N1(C(c2cc(CCC)[nH]n2)=O)CCCCC1C(C)NC(c1ccc(Cl)s1)=O CC1(F)CN(C(c2cccc3c2OCO3)=O)CCN(C(C2C3CCCOC23)=O)C1 N1(c2n(C3(C)CCOCC3)nnn2)CCC(F)(F)C(CNC(=O)C(N)=O)C1 c1(C(N2C(CNC(COC)=O)COCC2)=O)nc2ccccn2c1F N1(C(c2c[nH]c(=O)cn2)=O)CCOC2(CCN(C(=O)C3CC3)CC2)C1 C1(CC(=O)NC(CN(C)C(C2(CO)CC(C)(C)C2)=O)C2CC2)CC2(CCC2)CO1 C(=O)(CCCNC(=O)C(Cc1ccccc1)OC)NCC(COCC)OC N1(C(C(C)OCC(C)C)=O)CC(O)(C2CCN(C(c3sccc3CO)=O)CC2)C1 c1(C(=O)NC2CN(C(C3C(C)N(C)CC3)=O)C2)nc(C2CC2)ncc1Br CCCC(C(=O)O)N(C)C(C1CCN(Cc2cnn(CCF)c2)CC1)=O N1(C(c2cc(C)[nH]c2C)=O)CC2(CC2)CC1C(=O)NCC(C)(C)N(C)C C1(C(=O)NC(C#C)C2CCC2)CCCN(C(=O)CCCCC#N)C1CC CC1(C)OC2(C(F)F)CC1(C(N1CCC(NC(c3cncn3C3CC3)=O)C1)=O)C2 C1(C(N2CCC(CNC(C(c3ccccc3)N(C)CC)=O)C2)=O)C(C)(C)C1(F)F C1(C(N(CC(C2CC2)NC(CSCC)=O)C)=O)CCC1C(F)F C(=O)(C(C)P(C)(C)=O)OC.C(CC1CNC(=O)c2cc(on2)C(=O)N1)OC N1(C(CC2ON=C(C)C2)=O)CCC2(CC1)CCN(C(C1CCCC1CF)=O)CC2 N1(C(c2cc3ncccc3[nH]2)=O)CC2CCN(Cc3cc(F)c(Cl)cc3O)C2C1 c1(C(N2CC(N(C)C(C3(C#N)CCOC3)=O)C2)=O)ncc(F)cc1F c1(SC)nc(N(C(c2cn3ccccc3n2)=O)CC2(C)CNC2)nc(C)c1Br N1(C(c2c(C)cn(C)n2)=O)CCC2CC2(C(N2CCN(C)CC(O)C2)=O)CC1 N1(C(c2cccc(-n3ccc(C)n3)c2)=O)CCCCC(N(C)C(C2CC2C)=O)C1 c1(C(N2CC(C(C(=O)NC(CC(C)C)C)O)C2)=O)cccc(O)n1 N#Cc1cc(F)c(CNC(C2(C(F)(F)F)CCOC2)=O)c(F)c1 C1(NC(C(C2(O)CC2)OC)=O)CCN(C(C2(C)C=CCC2)=O)CC1 C1(OC)CCCCC1C(=O)N(C)CC1CCN(C(=O)C=CC=C(Cl)Cl)CC1 C1(NC(C(C)=C2CC2)=O)CCN(C(c2cn(C3CCC3)nc2C)=O)C1C N1(C(CCSc2c(C)cc(C)cc2C)=O)CCN(C(=O)C(C)C#N)CC2(CC2)C1 C1(C(N2CC(N(C(C(C)NC(=O)NC3CC3)=O)C)C2)=O)CC2(C1)OCCO2 CCC(C)CCCCC(=O)NCC1(C)CN(C(C2(C)CS(=O)(=O)C2)=O)CC1C CN1CC(C(=O)NC2(CCCNC(C3CC4C=CC3C4)=O)CC2)NC1=O c1(OC)ccccc1C(CNC(C1CC(C)(F)C1)=O)NC(=O)C(O)C(F)F N1(CC(=O)N(C2(SC3CC3)CC2)C)CCN(C(C2(C3CCCCO3)CC2)=O)CC1 CC1(C(=O)NCC2CN(C(C34CCC(C3)C4)=O)CCO2)CC2CCC1O2 CC(C)CC(CNC(=O)Cc1cnn(C)n1)NC(=O)CSc1nncn1C N1(C(Cc2nc(C)[nH]n2)=O)CC2COCCC2(NC(c2cc(C(N)=O)c[nH]2)=O)C1 CC(CC(C)NC(c1cc(N2CCCC2)ccn1)=O)N=c1[nH]nc(C2CC2)o1 Cc1cc(C(N2CCN(C3CN(C(C4(C(C)(F)F)CC4)=O)C3)CC2)=O)c(C)n1C C(CCC)(C(=O)NCCC1CCSC1)NC(c1c(CC)c[nH]n1)=O c1(C(=O)NC(CN(C(C2C(C)(C(=O)OC)C2)=O)C)C)nccn2c(Br)cnc12 c1(C(=O)NC(CC)CNC(c2cncc(C)c2Cl)=O)coc2c1C(=O)NCCC2 C1(CC(N2CC(C)C(NC(C3CCC(=O)N3C)=O)C2)=O)CCCC(C)(C)O1 CC(=O)C(C)CC(C)C(=O)NCC(CC(C)C)NC(c1cncn1C(C)C)=O C1(CC(=O)NCC2CCC(NC(C(C=C)(C)C)=O)C2)CC2CCC1CC2 C1(C(=O)NC(c2nn[nH]n2)CC)N(C(=O)C(CC2CC2)OC)CCCC1(C)C c1(C(C)(C)C)cc(N(CCCO)CCC)n2ncc(C#N)c2n1 c1(-n2cc(CN(C(c3cnc(CC)o3)=O)C)nn2)ccc(C)c(Cl)c1 c1(C(=O)NC2C(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CC2)cnn2c1OCC(O)C2 c1(N(C)C)cnc(C(=O)NC2CC2NC(=O)CCCn2ccnc2)nc1 c1(C(N2CCCC(c3cn(CC(COC)O)nn3)C2)=O)cc(C)nc(Cl)c1 Cn1c(C(=O)NC2(C)CCN(C(=O)CC3CCCCC3(F)F)C2)cc2occc12 N1(C(C(CC)F)=O)CC(NC(=O)CCc2csnc2C)C(C)(C)C1 C1(Cl)(C(=O)NC(C)CNC(c2cnn(CC(F)F)n2)=O)CC1(C)C c1(CCC(=O)NC2CCC(Cn3cc(CN4CCOCC4)nn3)C2)nc(=O)o[nH]1 c1(C(C)C)ncc(Br)c(N2CC(N(CCN(C(=O)C(F)(F)F)C)C)C2)n1 c1(C(=O)NC(C(=O)N(CC)CC2CC2)C)ccnc(-n2cccc2)c1 CC(CC#N)N=c1[nH]c(=NC(CCO)c2ccccc2Cl)c2cc(F)cc(F)c2[nH]1 C1(NC(c2c(CC)c[nH]c2)=O)CC12CCN(C(C1CCC(=O)O1)=O)C2 C(=O)(C1COc2ccc(Cl)cc21)NC1CC(C)(NC(c2cccn2C2CC2)=O)C1 C1(CC(=O)NCC2(CNC(=O)CC3CC(F)C3)CC2)CCCC(F)(F)C1 c1(CC(=O)NCC2CN(C(=O)Nc3scnc3C3CCCC3)C2)ccccc1Cl c1(-c2cccc(C)c2F)nc2c(s1)CCN(C(C1CCC(CO)CC1)=O)C2 c1(C(=O)NC2CC2CNC(C2(F)CC23CCCCC3)=O)c(F)cccc1Br C1(CC)CN(C(=O)C(COC)COC)CC1NC(c1ccc(NC(C)=O)cc1)=O CC1(C)CCOC1CNC(C1CC(NC(C2CCN2C(C)(C)C)=O)C1)=O c1(C(N(CC(C)NC(=O)CC(F)(F)F)C)=O)cc(Br)c(F)cc1F c1(CC(=O)NCC2C3CN(C(=O)CCCC(F)F)CC23)cccc(F)c1F C1(NC(C2CN(C(c3cc(Cl)ccn3)=O)CCC2O)=O)CCc2ccccc2C1 Cn1cnc2c1CCCC2C(=O)NCC1(F)CCN(C(C2CC(F)(F)C2)=O)C1 c12cccc(n1)CC(=O)N2.c1(CCC2(C(=O)OCC)COC2)ccccc1F N1(C(c2ccc(CC)c(F)c2)=O)CCCC(C)(C)C1CNC(=O)C1=CCOCC1 N1(C(C2(SC)CC2)=O)CCC(NC(=O)C(n2cc(C)cn2)C)C1 C(=O)(C(C(C)C)NC(=O)CC=Cc1ccccc1)NCCNC(C(C)(C)SC)=O C1(NC(COC)=O)CCOCC1NC(c1cccc(-n2cc(C3CC3)nn2)c1)C C1(CC#C)CN(N2CCN(C(=O)C(c3ccc(OC)cc3)(F)F)CC2)C1 C(=O)(C(C)(C)CCC#N)N1CC(OCCC(=O)NCc2ccc(CC)s2)C1 CCN=c1[nH]c(C(=O)NC2CC(F)CN(C(=O)C(C)Sc3ccccn3)C2)cs1 c1(NC(C(C2CCN(C(c3c(F)cccc3F)=O)CC2)C)=O)cc(F)cc(I)c1 S(=O)(=O)(c1cccc(S(C)(=O)=O)c1)C1N2C(C)C(CC2)C1 N1(CC(=O)NCc2ccc3nc[nH]c3c2)CCC(=C(F)F)CC1 C1(NC(C(C)C2CCCC2)=O)CC2(C1)CC(C(=O)NOC1CCOC1)C2 c1(C(CNC(=O)C(=O)NC2CCC2)OC)cccc(O)c1 C=CC1OCCCC1C(=O)NCc1cn(CCNC(=O)C(CC)C(C)C)nn1 C1(CNC(CCN(CCC)C)=O)CN(C)CCN1C(=O)CC1COC(=O)C1 C1(C(=O)NC(CC(C)C)CNC(C2COC(=O)N2)=O)CC2CC1C1CC21 C(=O)(CCCCCCC(=O)C(CCC(C(C)C)OC(C)=O)=O)OC.N1CCCC(=O)C1 C=CCC(C(=O)NC(CNC(=O)C=CC(C)C)CC(F)(F)F)C(C)C C1(NC(=O)Cc2cccs2)CC2CCC1(CO)C2.C12C3CC4C(C3)C14C(=O)N2 Cn1nc(C(C)(C)C)cc1C(=O)NC1COCCC1NC(=O)CC1CCOC1 N12CCOC(C1)C(=O)NCC2.c1(CCC(=O)NC2(CSC)CCC2)nc(C)cs1 c1(C(N2C(CNC(c3n(CCC)ncc3)=O)C(C)CC2)=O)cc2n(c1)CCSC2 c1(CC)ccc(C(=O)NCC2(OC)CN(C(C3(F)CCCOC3)=O)C2)cc1 c1(OC)nsc(C(c2nnnn2Cc2ccco2)NC2CCC(F)(F)C2)c1Cl CCC(COC)N=c1cc(C)[nH]c(=NCC2CCOC3(CCC3)C2)[nH]1 C(=O)(CCC1CCc2ccccc21)N1CC(NC(Cc2cnc(C)s2)=O)C(C)C1 C1(NC(c2n(C)nc(C3CC3)c2)=O)CCCC(NC(=O)C(F)=CC2CC2)CC1 N1(C(C)=O)CCC(C(CO)N(C(=O)C(=O)NC)CC)CC1.C(C)(C)(C)NC1CC1 C1(SCC(=O)NC(C2CC(NC(C3CCSCC3)=O)C2)C)CCCC1O CCC(C)C(C(=O)NC1CC(NC(c2nnn(C)c2C(F)F)=O)C1)NC(=O)OC c1(C(c2n(CCC)nnn2)NCC(C)(C)OCC2CC2)nc(F)ccc1Cl c1(CC)cc(C(=O)N(CCC(=O)N2CC(N3CCCC3)C2)CC)nn1C C1(NC(C2CC23CCC3)=O)CC2CN(C(=O)CN3CCCNC3=O)CC12 C1(CNC(c2c(C)con2)=O)CC(C)(C)CCC1NC(c1cccn(C)c1=O)=O C1(CNC(C2CCN(CC3CC3)CC2)=O)CCN(C(C2(O)COC2)=O)CC1 C(=O)(CS(=O)(=O)C1CCCN(C(C2(O)CC2)=O)C1)OCC CCC(CC(F)F)C(=O)NCC1(NC(c2ccc(CC)cc2)=O)CC1.C1(SC)CC1 C(C(O)C(=O)NC(C)(C)CCF)NC(C1(NC(C)=O)CCC1)=O c1(C(N2CC3C(CNC(CNC(CCCCC)=O)=O)(C3)C2)=O)ccc(N)cc1F N1(C(C(=O)Nc2cnn(C(F)F)c2)=O)CCN(Cc2cccc(F)c2)C(=O)C1 c1(CC(NNc2ccc(C)cc2)=O)cnc(=NCCC(F)(F)C(C)O)[nH]c1 c1(N(CCC)C)ccc(C(=O)NCCC(C)N(C(=O)CN2CCCC2=O)C)cc1 C1(N(C(C=CC=CCC)=O)CC)CCCN(C(c2cnn(CCO)c2C)=O)CC1 C1(NC(c2c(C)cc(F)s2)=O)C2CC3C(C2)C13C(=O)NC1(C)CCCC1C n1(C(C)(C)C)cnc(C(=O)NCC2CC(CNC(c3ccsn3)=O)CO2)n1 c1(NC)cnccc1C(=O)NC(CNC(c1ccc(C2CC2)s1)=O)C1CC1 c1(OC)c(C(=O)N(C)CCOCCNC(C2CC(F)(F)C2)=O)c(C)nn1C N1(C(C=C(CCC)C)=O)CC2(CCC2)CCC1CNC(=O)CC1CCC(O)C1 N1(C(C2=C(CC)OCCC2)=O)CCCC2(CCN(C(c3nc(Br)c[nH]3)=O)C2)C1 C1(C(N(C(C)C)CCc2ccccc2)=O)CC2CCC1N2 CC1CCC=C1C(=O)NCC=CCNC(c1sc(C2CC2)nc1C(C)(C)C)=O C(=O)(C1CC(=O)Nc2cc(F)ccc21)NC1CC(NC(c2onc(C)c2C)=O)C1 c1(C(=O)NC(CN(C(C(CC)OC)=O)C)(C)C)cc(N(C)C)nc2ccccc12 C(C)(C(=O)NC(CNC(C)=O)CC(=O)N)OCC.C(C(F)F)(C1(C)CC1)OC.C1CO1 c1(CCC(=O)N(C2CC(NC(CSC)=O)C2)C)n[nH]c(=N)s1 C1(C(C)C)CCN(CC(=O)N(CCN2CCCC2)CC2CC2)CC1 CC1(C)CCOC1CS(=O)(=O)NCc1sccc1Cl CCC(C)(C)C(=O)N1CCCC(C(C)(O)CNC(c2ccc(OC)nc2)=O)C1 c1(CCC(N2CC(C(N)=O)(CNC(CC3C(C)C3)=O)C2)=O)c(F)cccc1Cl c1(NC(C(=O)NCCc2ccc(CNC)cc2)=O)nccc(Cl)c1Cl C12(C(N3C(C)CC(NC(=O)CCc4cncs4)C3)=O)CC3CC(C1)CC(C)(C3)C2 c1(C(=O)NC2C(CNC(C(C)(C)SC)=O)C2)cc(C)n(-c2ccccc2)n1 C1(CCNC(C(SC)SC)=O)CCN(C(c2nnc(C(C)C)s2)=O)CC1 c1(C(=O)NCCN(C(CC2(CC)CC2)=O)C(C)C)ccc(N)c2ccncc12 C(=O)(C1CCCc2ncnn21)NCCOCCNC(C1CCCC(C)C1)=O N1(C(Cc2c(SCC)cccc2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)C(C)C1 N1(C(C2N(CCC)CCC2)=O)CCCCC1CC(N1CC2CC1C2)=O n1(CC(=O)NC(C2CCCC2)CNC(C(C)NC(CC)(C)C)=O)ccc(C)n1 Cc1ccn2cnc(C(=O)NCC3(O)CCCN(C(=O)C(O)C(C)C)CC3)c2c1 C(=O)(C1=CCS(=O)(=O)C1)NC1C(NC(C2(C)CCC(C)CC2)=O)CCC1 c1(NC(=O)Cc2cc(F)ccc2Br)cnn2c1CNCC2 N#Cc1[nH]c(=NC2CCC3CN(C(C4Cc5cscc5C4)=O)CC3C2)sc1Cl Cc1ccc(C(=O)NC(C)CCC(=O)NC(c2cccnc2)CO)cc1 C(C(CC(C)C)C(=O)NCC1(CN(C)C)CCCCC1)NC(CC=C)=O C1(CCOC)CN(C(=O)CCCN(C)C)CCN1C(c1cncs1)=O CCC(C)(C(=O)NCCC(CNC(=O)C(=O)NCC(F)F)OC)C(N)=O N12CCC13CCCN(C3)C(=O)CC2=O.c1(NC(NC(C)C)=S)cnccc1F N1(C(c2ccc(CC)cn2)=O)CC2COCCC2(NC(C2SC(=N)NC2=O)=O)C1 C(=O)(C(C(C)(C)C)OC)NCC1CCCC(NC(CCCOCC=C)=O)C1 C1(NC(C2CC(=C)C2)=O)CS(=O)(=O)CC1NC(=O)COc1cc(F)ccc1F C1(CC)CCN(C(c2cncs2)=O)C1C(=O)NCCOCCOC N1(C(Cn2c(C)nnn2)=O)CCC(C2CCN(C(c3cc(C(N)=O)co3)=O)C2)C1 N1(C(C(C)(F)F)=O)CC2CCC(NC(=O)CC(O)CC3CC3)C2C1 c1(C(=O)NC(C)(C)CCNC(C2C3CCC23)=O)cc(F)cc(F)c1O CCCCCCC(C)(CCC)C(=O)NC1(CCCNC(C2(C3CC3)CC2)=O)CC1 c1(CC)ccc(C(=O)NC(C(=O)N(C)Cc2nccn2CC)C2CCCC2)s1 c1(C(=O)NC(CNC(Cc2c(OCC)nccc2)=O)C)c(F)ccc(OC)c1N CC(N=c1nc2scnc2c(N2CCCC(n3ccnn3)C2)[nH]1)c1ncc[nH]1 C1(NC(CC2(OC)CCC2)=O)C2CCN(C(c3ccoc3Br)=O)C12 N1(C(c2scc(CNC(C(C=C)(F)F)=O)c2)=O)CC2CCCC(O)C2C1 N1(C(c2c(C(C)C)cco2)=O)CCOC2CN(C(C3CC3C(N)=O)=O)CC12 CC1CN(C(c2coc(C#N)c2)=O)CC(CCNC(c2c[nH]nc2F)=O)O1 NS(=O)(=O)CCCC(=O)NC1CCC1NC(C1CCc2nc[nH]c2C1)=O c1(C(=O)NC2CC(CCNC(CCc3cc(N(C)C)no3)=O)C2)cc(N)ccn1 c1(C(=O)NCC23C(CN(C(C4CC5C=CC4C5)=O)C2)C3)ccc(F)c(Br)c1F C12(C(=O)NC(C3CCN(C(C4(C5CCC5)CC4)=O)C3)C)CCCC1CC(=O)CC2 C1(NC(=O)CCN(CCCO)C(=O)Cc2nc[nH]n2)CN2CCCC1C2 C1(NC(C2C(C(C)C)C2)=O)CCN(C(c2csc(-c3nc[nH]n3)n2)=O)C12CC2 CC(O)(C(=O)N1CC2C(C(=O)Nc3cc(I)ccc3I)C2C1)C(F)(F)F C(=O)(CCCC(F)(F)F)NCCC1(C)CCN(C(c2cc(CC)oc2C)=O)C1 C1(CNC(=O)C=Cc2cocn2)CCC2(CN(C(C3(O)CCOC3)=O)C2)O1 C12COC3(CC1C3)C(=O)N2.C1(CC(=O)NCCCNC(=O)NC)CC12CC2 CC1=NS(=O)(=O)N(C)C=C1C(=O)N1C2CCC1CN(C(C1CC(N(C)C)C1)=O)C2 CCC(C)(CC)C(=O)NCCC(O)C(=O)N(C)CC1CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NCCC(C)NC(c1c(C)ccnn1)=O N1(C(c2nc(CC)oc2)=O)Cc2n[nH]cc2C1C(=O)NC1CC(CSC)C1 C1(NC(c2occ(C)c2)=O)CCC12CCN(C(c1ccc(N)c(Br)n1)=O)CC2 c12occc1CN(C1CC1)C2=O.n1(C2(C(=O)NC3CC3(Cl)Cl)CC2)cncn1 C(=O)(CCC(=O)N1CCC(NC(C2C3CCC23C(=O)O)=O)C1)NCCCOC C1(C(=O)NCCCN(C)C)(NC(C2OCCN(C(C)C)C2)=O)CCC(F)(F)CC1 C=C(C)C(C)(C)C(=O)N1CC2(C1)CN(C(C1(C)CC(F)C1)=O)C2 N12CC3CCN(CC3C1)N(C)CC2=O.C1(C(=O)OC)C2CCC1(C(=O)O)C2 C1(NC(CC(=C=C)C)=O)CN(C(=O)CCc2cccc(Cl)c2Cl)CC12CC2 CS(=O)CCC(=O)NC(C1CCN(C(=O)CCc2ccncn2)C1)(C)C N12CCN(CC1)C(=O)C(C1CCCC3CC13)N1CCC2C1.C1(C(O)C2CC2)CC1 c1(CNC(c2ncn(C)c2Cl)c2n(CC(=C)C)nnn2)c(Cl)n[nH]c1C N1(C(c2c(C)occ2)=O)CCC(NC(c2ncsc2S(N)(=O)=O)=O)CC(C)(C)C1 N1(C(C2CCN(C)C2=O)=O)CC2CCC(C1)N2C(c1nc(=O)n(C)[nH]1)=O C1(O)(CN(C(c2c(C)onc2)=O)C)CCN(C(=O)CN2CCCC2=O)C1 c1(C(=O)NCCN(C(c2nc(CC)sc2)=O)CC)cc2ccc(F)cc2nc1O Cc1cc(Cl)ncc1C(=O)NCCN(C1CCCCCC1)C(c1nccn1C)=O c1(C(=O)NCC2C(C(=O)NC(CC=CC)CO)CC2)ccnnc1O N1(CCC(=O)NCCC(C)NC(C2CC3(C2)CC3F)=O)CCCCCC1 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CC(NC(=O)CCCCC)CCC1C CC1Cn2nc(C(=O)NCC3CCN3C(c3ccc(Br)o3)=O)cc2C(=O)N1 N1(C(c2cn(C)nc2O)=O)C2COCC1CC(NC(=O)CN1C(=O)CNC1=O)C2 N1(CC)CCCN(C(C2(C(C)C)CCN(C(c3c(C)cccc3C)=O)C2)=O)CC1 Cn1nc(C(=O)NC2CN(C(C3CCCOCC3)=O)C2)c2c1CCC(C)(C)C2 C12(CN(C)C(C3CCCCN3S(=O)(=O)c3cccs3)=O)CCC(C#N)(CC1)CC2 C12(C(=O)NC(CC)CNC(=O)CCC(=O)N(C)C)CC3CC1C2C3O.C1CCO1 Cc1cccc(C(N2CCC3C(NC(C4CN(C)C4)=O)C23)=O)c1Cl C1(NC(C2C(C(=O)OC)C2)=O)CN(C(c2ccnc(OC(F)F)c2)=O)CC1(C)C c1(SCC)ccc(C(=O)NCC2C=CC(NC(=O)CN(C)CCO)C2)cn1 C(=O)(C(C)CS(C)(=O)=O)NCc1c(CCNC(c2ccc(C)nc2C)=O)ocn1 Cc1ncccc1CC(N1CCCC1CCC(=O)NC(c1cnc[nH]1)C)=O c1(C(=O)NCC2OCCC(NC(C=C(CC)C)=O)C2)c(C(F)(F)F)cccc1F C(CC(CC)C(=O)NCCC(C)N(C)C(c1cnc(O)n1CC)=O)=CC C(=O)(C1COc2ccc(Cl)cc21)NC12CN(C(c3nc(C)sc3)=O)C(C1)C2 N1(CC(=O)Oc2ccc(C(CC)(F)F)cc2)CCCCC(=O)C1=O C(=O)(C(C)C(O)C(C)C)N(CC1CCN(C(c2scc(COC)c2)=O)CC1)CC N1(C(CC2CC(NC(C(C)CCN(C)C)=O)C2)=O)CCOCC(C)(O)C1 CC1CC(NC(=O)C(C)(C)C)CN(C(=O)CCSc2ccncc2Cl)C1 c1(CNC(C2CCC(F)C2)=O)ccc(C(=O)NC2CC(F)C2)nc1 CCCCN=C(NCC(C)(C)C)NC1CCOC(c2cccc(Cl)c2)C1 c1(C(=O)NC(CCN(C(C2=C(C)OCC2)=O)C)C)cc2c(nc1O)CCCC2O c1(C(C)(C)C)cc(NC(=O)NC2CCOC2c2ccccc2)n(CCO)n1 CN1CCCCC1CC(N1CCCC1Cc1ccccc1)=O C1(CC)CN(C(=O)C=C(CC)CC)CCC1NC(=O)C(=O)NCC(F)F C(=O)(C(CC)C(=O)N1C(CO)CCC1C)OCC.CC(=O)O CCCCC(C(=O)N1CC2CC1CN2C(=O)CCOC)NC(N)=O Cc1cccc(C2CC2NCCNC(=O)C(c2ccc(C)s2)O)c1 C1(C(=O)NCCCCCNC(c2c(CC)ncs2)=O)CCN(S(=O)(=O)N(C)C)C1 CCC(CC(=O)N1CCC(N(C)C(c2cc(OC)cnn2)=O)C1)CC(C)C c1(CCC(=O)NCC(C)NC(CC=CCC)=O)cccc(C(=O)OC)c1 N1(C(CN2C(C)CC2)=O)CCCC(C(=O)COC(=O)Cc2cc(C3CC3)no2)C1 C1(C(N2CCC(CNC(C(C)c3ccco3)=O)CC2)=O)CC2(CCCCC2)C1 C(=O)(C1CCc2cccnc21)N1CC2CC(NC(=O)CC3CSC3)CC2C1 c1(C(N2C(C)CC(NC(C3(CCC=C)CC3)=O)C2)=O)cnnc2ccccc12 C(=O)(C(C)(C1CC1)NC(=O)C(C1CCC1OC)NC(C1CCOC1C1CC1)=O)OC N1(C(CCC)=O)CC2(CC(NC(=O)C(F)C(F)(F)F)CO2)C1 c1(C(N2CCC(C(C)NC(c3ccc(C(N)=O)cc3)=O)C2)=O)cccc(=S)n1O C1(CCNC(c2cccnc2S)=O)CC(F)(F)CN1C(=O)Cc1cncnc1 C1(NC(C2CC(CCC)C2)=O)CCC(CNC(=O)Cn2cc(C(F)F)cn2)CC1 O=C1c2ccccc2C(=O)N1CCS(N1CC2(CCC(=O)O2)C1)(=O)=O c1(N(CC(CN(C)C(c2n[nH]c(C3CC3)n2)=O)O)C)ncc2c(ncn2C)n1 C1(COC)(NC(C2CNC(=O)C2)=O)CN(C(=O)CCn2cncn2)C1 O=C(CS(=O)(=O)c1ccc(Br)cc1)NC1CCN(C(c2ccc[nH]2)=O)C1 C1(C(c2ccccc2)C)CN(C(=O)CC2(C)CC2)CCN1C(c1scnc1C)=O c1(CC(Cn2ccnc2C(C)=O)OCOC)ccc(F)cc1F CN1CCN(C(=O)CCOC2CCCC2)C(C(N2CCC2(C)CCO)=O)C1 Cc1ccnc(C(N2CC(CN)C(C)C2)=O)c1Br CC1CCCCC1(CNC(=O)Cc1n[nH]c(=N)s1)NC(=O)C=C1CCCC1 c1(OC)c(C(=O)NC2CC(C)(CNC(=O)Cc3cncs3)C2)ccnc1Cl C(C(CCC(=O)O)C(F)(F)F)NC(C#C)CC1CCCO1 c1(NC(=O)CCCF)ccc2occc2c1.C12CCC(CC1)NC2=O c1(OC)cc(CNC2CCC(C)C(C)C2)ccc1O C#CC1(O)CCN(C(=O)C(Cn2cccn2)NC(=O)C(C2CCCC2)OCC)C1 C1(NCCNC(C(C)N(C(=O)C(C)Cn2cccn2)C)=O)CCOCC1 N1(C(Cc2cnc(C)s2)=O)CCCC(NC(C2COCC2C(N)=O)=O)CC1 C12(NC(c3cc(O)nc(O)n3)=O)CCC(C1)N(C(c1nc(Cl)ccc1Cl)=O)C2 CCC(CC(C)C)C(=O)NC1COC2(CNC(c3cocn3)=O)CC1C2 C(CC(C)CC)(C(=O)NC(C)CCC=C)NC(c1c(C#C)cn(C)n1)=O C#CCCC(O)C(=O)N1CCC(CC(C)NC(c2ccc(C3CC3)nc2)=O)CC1 C1(C(C)C)(CC)CCCN1C(C1C(C=CC)CN(C(=O)COCCCOC)C1)=O CCC(C(=O)NC(C)CC1CCN(C(=O)Cc2ccc(O)cc2)CC1)C(F)(F)F Cc1c(C(=O)NCC(C2CCN(C(=O)C=C3CCN(C)C3)CC2)C)cccc1F C(=O)(CCCN=c1nccc[nH]1)NCC1N(C)CCN(C(=O)CCC(C)(C)F)C1 c1(C(=O)NCCN(CCOC)C(c2nc(C3CC3)no2)=O)nc(Br)c[nH]1 C(=O)(CC(=O)N1CCCC1C1(NC(c2c[nH]cc2CC)=O)CC1)NCC c1(NCC(c2ccccc2)C)sc(CC(=O)O)cc1C#N c1(C(N2CC(F)(NCCNC(CSCC#C)=O)C2)=O)c(OC)cccc1OC N1(CCC)CC(C(N2CC(N(C(C3C4CC5C(C4)C35)=O)CC)C2)=O)CC1=O c1(C(=O)NCC2(CCNC(C(C)C3CCOC3)=O)CC2)ccc(P(C)(C)=O)o1 c1(CCNC2C(NC(=O)OC(N(C)C)=O)COCC2)cccc(Br)c1 C(=O)(C(C)(C)CC(C)(C)C)NC1CC(NC(C2(COC)CCCO2)=O)C1 N1(C(C(=Cc2ccco2)C)=O)CCC(C)(C)C(C(=O)NCC(C)(C)CC(C)O)C1 C(=O)(CC(C(C)C)C(C)C)NC1CCCC(CNC(C(C)(C)SC)=O)C1 Cc1ccc2c(c1)c(CCNC(=O)Nc1ccc3nc(C)sc3n1)cn2C c1(CC)cc(OC)cc(C(=O)N(CCNC(=O)CN2CC3CC3C2)C(C)C)c1 c1(C(=O)NC2C3CN(C(CCCNC(C)=O)=O)C2C3)c(F)cccc1Br C(=O)(C1=CCCCC1C)N1CC2C(NC(c3c(C)cn(C(C)C)c3)=O)(C2)C1 C1(NC(c2c(C)nn(C)c2)c2nnnn2Cc2ccccc2)C(O)C2CCOC12 N1(C(CN(C(C)=O)C)=O)CCC2CC2(C(=O)NCCCC(C)CO)CC1 N1(C(c2c(C)ccnc2)=O)CC2CCCN(C(=O)C(F)(F)CF)C2C1 C1(NC(c2c(C)cncc2)=O)CC2C1CCN2C(=O)CN1C(=O)CNC1=O N1(C(C(C(C)C)F)=O)CCC2CCC(C1)N2C(C1(C2CCC2)CC1)=O Cc1nccn1C(C)C(=O)NCC1CC(O)(CNC(=O)CSc2cccs2)C1 C1(NC(c2c(CC)onc2)=O)CCN(C(=O)C(c2ccccc2C)C)CC1CC C1(CNC(Cn2nc(C)n3c2ncc3)=O)CC2CCCC2N1C(C1CSC1)=O C1(Nc2ncc(C)cn2)CCCN(C(c2cnc(-c3ccco3)s2)=O)CC1 C1(O)(CC(N2CC(OC3CCN(C(CCCC=C)=O)CC3)C2)=O)COC(C)(C)C1 Cc1[nH]nc(C(=O)NC2CN(Cc3c[nH]nc3C3CC3)CC2n2ccnn2)c1Cl Cn1c(=O)ccn(CC(=O)NC2(CNC(c3csc4cncn34)=O)CCC2)c1=O c1(C(=O)NCCC(C(=O)NC(C2CCC2)C)O)n[nH]c2c1CCC2 N1(C(c2cn(CCC(C)C)nn2)=O)CCN(C(c2cnnn2C)=O)C(C(C)C)C1 c1(SC(C)C(=O)NCC2CCCN2C(=O)CN2CCSCC2)ccccc1F C1(C(N2C(C(=O)NC(C(=O)NCC)C)C3CC3C2)=O)CC2(C1)CC21CC1 C1(C(=O)NCC(=C)F)CCCCCN1C(=O)Cc1cnns1 N1(C(CC2CC(OC)C2)=O)CCCCC(NC(=O)C(F)(F)CO)C1 N1(C(c2cccc(OCC#C)c2)=O)CCN(C(C2(C#N)CC(C)C2)=O)C2(CC2)C1 C1(C(N2C(CN(C(CC(C)(F)F)=O)C3CC3)CCC2)=O)CCCC12CCC2 N1(C(c2c(CC)nc(=N)[nH]c2)=O)CC2(C1)SCCC2NC(c1cnc(C)s1)=O C(C(CC(=O)N=c1cc(C(N)=O)n(C)[nH]1)NC(c1cccc2c1CCC2)=O)OC Cc1nc(C)c(C(N2CCCC2CNC(c2cccc(Br)c2Cl)=O)=O)nc1C C(C1Cc2ccccc21)NC(C(C)CCN(C)C)=O.C1C#CC(=O)N1 C1(C(N2CC3CC(C)C3C2)=O)CC12CCN(C(C1COCC1(C)C)=O)CC2 c1(C(N2CCC(=CCNC(C(C)=O)=O)CC2)=O)cccc2c1OCCO2 C12(CC(=O)NCCC3CC(NC(=O)CCc4nncs4)C3)CCCN1CCC2 C1(C(CC)NC(=O)N(CCO)Cc2ccncc2)Cc2ccccc2C1 c1(C(C)OCC)nc(-c2ccsc2C)n(C(C)C(C)C)n1 c1(CCC(=O)N(CCC(C)NC(C2CCC(CCO)CC2)=O)C)ccc(F)nc1 c1(C(=O)OC)cccc2c1OCCN2C(c1ccc(Cl)cc1Cl)=O c1(C(=O)NC(C(C)NC(=O)CCCN2CCCC2)C)ccc[n+]([O-])c1 C(=O)(CC(C)(C)C(F)F)NC(C(C)NC(=O)CNC=O)CO c1(C(C(N2CCC(CSC)C2)=O)NC(COCCCC)=O)c(C)cccc1Br C1(C2CCN(C(C3(Cl)C(C)(C)C3)=O)C2)CCCCN1C(=O)COc1ccccc1 c1(C(N2CCCC(CN(C(C(C)CF)=O)C)C2)=O)cc(Cl)c(F)cc1Cl C(C)(C(=O)NCC1CCC1NC(C1(CC(F)F)CCC1)=O)=CC C#Cc1ccc(C(N2CCCC(O)(CNC(c3ccnn3CC)=O)C2)=O)c(C)c1 N1(C(C(CCC)C)=O)CCN(C(=O)CNC(=O)Nc2ccco2)C2(CCC2)C1 C1(C(=O)OC)CC1CCCNCCN(C)C.C1(=O)CN1C1CC1 C1(C(=O)NC(C2(CNC(c3n(C(C)C)ccc3)=O)CC2)C)CCCC12CC2 N1(C(=O)CC2CC(O)CN2C(=O)C2CC2)C2CCC1CC1(CC1)C2 N#Cc1ccc(F)c(F)c1N(C(C1=CC(C2CC2)=CC=Cc2ccccc21)=O)C1CC1 C#Cc1ccc(CC(=O)NCC2(C)CC(NC(=O)CCS(C)=O)C2)cc1.C1(C)CC1 CC(C)C(CC(=O)NC(c1cncn1C)=O)NC(=O)Cc1cn(CC(N)=O)nn1 CC(C)CC(C)(O)C(=O)N1CCN(C(c2ccoc2Cl)=O)C(CS(C)(=O)=O)C1 N1(C(CC(C)(C)C2CC2)=O)CCCC12CCN(C(=O)C(O)C1=CCCCC1)C2 N1(C(=O)NCC(c2ccc(Br)cc2)OC)C2CCCC1CN(C)C2 C(=O)(C(C)(C)C(=O)N1CCOCC1)N(CC(C)(C)CNC(C1CCC(=O)C1)=O)C C1(C(=O)NCCn2cc(COCC(C)O)nn2)CC2CCC1C2 C1(NC(Cc2ccn(CC)n2)=O)CCCCN(C(c2cnnc(C)c2)=O)C1 c1(C(=O)OCCC(N2CC(OC)CC(CC)C2)=O)cccc2oc(C)nc12 N1(c2ccnc(OC)n2)CCC(C2CCN(C(c3cc4n(n3)CCC4)=O)CC2)C1 c1(C(N2C(C(C)(C)NC(=O)CC34CCCC3C4)CCC2)=O)ccc(C2CC2)nc1 N1(C(=O)Cc2ccoc2)CCC2(CCCN2C(=O)CSc2n[nH]c(O)n2)C1 c1(C(N2CCCC(NC(=O)NC3CCCC3)C2)C(=O)NCC)ccc(F)c(F)c1 C=CC(F)(F)C(=O)N1C(CNC(=O)Cc2cccnc2O)CC2CC12 c1(C(=O)OC)ncc(NC(=O)NC2C(CC=C)C(O)C2)cc1F C=CC1CN(C(C2COCC(=O)N2C(=O)OC)=O)CC1NC(=O)OC(C)(C)C c1(C(=O)NCC2CC(NC(C3(CCOC)CC3)=O)C2)cccc(C#N)c1 N1(C(C(CC=CC)CC)=O)CCCN(C(=O)COCCF)CC1c1ccccc1 c1(C(=O)NC(CC(C)C)CNC(=O)CC2CCC(O)C2)nc2ccccn2n1 C1(C(=O)NC(COC)C2(C)CC2)CC(O)CN1C(=O)CCC1CCCN1C c1(-c2cn(CC(N3CC(CCC)OCC3)=O)nn2)ccc(N)c(CC)c1 N1(C(C2CC(=O)NC(=O)N2)=O)CCc2ccc(C(=O)NCC3CCCO3)nc2C1 C(=O)(N1CCC(C(=O)NC2(C)CCSCC2)O1)C1N(C)C(=O)CC1 Cc1cc(CN2CC(F)CC2C(N2CCC(O)C(C)C2)=O)c(F)cc1Br N1(C(Cn2c(C)ncc2)=O)CCC(C)C(NC(c2cc(C(N)=O)cc(F)c2)=O)C1 c1(C(=O)NCC(CNC(CSc2n(C)ccn2)=O)(C)C)cccc(P(C)(C)=O)c1 N1(C(C(C)=C2CC2)=O)CC(C)(C)CC1C(N1CC(C(C)(C)O)C1)=O CC1CN(C(=O)CC2(O)CCCCC2)CCN1C(C1CC(C)(C)CN1C)=O C1(C(=O)NC2CC3(C2)CN(C(C2(F)CC2)=O)C3)CCc2nc(C3CC3)[nH]c2C1 CC1=C(C(=O)N2CC(C(O)C(=O)N(C)Cc3ccc(F)cc3)C2)CCCO1 n1(CCC(N2CC(CNC(c3cnc(=N)[nH]c3)=O)C2)=O)cc([N+](=O)[O-])cn1 c1(C(=O)NC(CNC(c2c(CC)n(CC)nn2)=O)C)cc(C)nc(O)n1 C=CCC(CC=C)C(=O)N(C(C)(C(=O)N(C1(c2cc[nH]n2)CC1)C)C1CC1)C N1(C(C2CCC(COC)C2)=O)CC2(CC2)CC1CNC(c1cn(C)c(=O)cn1)=O N1(C(C=CC2CCN(C(C(CCCC)=O)=O)CC2)=O)CC(C)(C)OCC1(C)C c1(C(=O)NCc2ccsc2Br)cnc2c(-c3ccc4nccn4c3)cnn2c1 N#Cc1cc(N2CCC(NC(=O)C=C(Cl)Cl)CC2)nc(-c2ccccc2)n1 CCC(C)(C)CCCC(=O)NC(CC(=O)NCCC(O)C(F)(F)F)C(C)(C)C c1(SC)cn(C)nc1C(=O)NC1CN(C(=O)Cc2cnccn2)CC1O C#CC1CC2CCC1N(C(C1(NC(=O)Cc3ccsc3C)CC(O)C1)=O)C2 Cc1cccc(NCC2(N(C(c3ncc[nH]3)=O)CO)CCOCC2)c1.C1CC(=O)N1.CC C1(C(N2CCC(N(C(=O)CCSC(F)(F)F)CC#C)C2)=O)CCCC(OC)C1 C12(C(=O)OC)CCOCC1CN(C(=O)Cn1cnc(C(=O)O)c1)C2 C(=O)(C(C)(F)C(=O)NC(C)CNC(C1CC1Cc1cncn1C)=O)OC CC(C)C(O)C(C)C(=O)NCC1(C)CCCN(C(c2cn3ncccc3n2)=O)C1 N1(C(CN(C2CCSC2)C)=O)CCC2(CC(C(=O)NC3CCCCC3)C2)C1 c1(C(N2CC(NC(c3nc(C)sc3)=O)C2)=O)cnc2c(c1)c(C)nn2C(C)(C)C C1(O)(CC)CCCN(C(=O)C(C)(CO)NC(C2COCC2C(N)=O)=O)C1 C1(OC)C(OC)CN(C(C2CCCOCC2)=O)C1CNC(=O)CC1CC1 N1(CC)CC(C)(C)C12CCC2.N1(C=O)C(CO)C(CO)C1CO c1(N2CCO2)ccc(I)cc1Br.NC(=O)C1CC1 N1(C(Cc2cn(C(C)C)nc2)=O)CC(NC(=O)CO)CC(O)C1 C(=O)(C(=O)NNC(=O)c1ccc(NC(c2csc(Br)c2)=O)cc1)OC c1(C(N(CC(C)NC(=O)Cc2ccc(F)cn2)C)=O)cnn(C)c1N C#CC1(C(N2CCC2C=C)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 C#CCCC(O)C(=O)NCC(O)CCNC(=O)CC1CCC(C)CC1 N1(NC(=NCC2CCCCS2)NC2CCCC2)CCCN(C(=O)CSC)CC1 N1(C(CCc2cn(C)nn2)=O)CCCC1(C)CNC(C1CC1OC(C)(C)C)=O C(=O)(C(C)(C)CCC(=O)NC1CCCN(C(=O)C(O)CC(F)F)CC1)OC N1(C(c2ccc(C(=O)NC)nc2)=O)CC2CC1CC2NC(=O)C=C(C)C(F)(F)F c1(CSCC)cccnc1C(=O)NCC1CC(CNC(c2c(C)noc2N)=O)C1 C1(CCNC(c2c(CC)cno2)=O)CC(F)(F)CN1C(=O)C=Cc1ccc(C)o1 N1(C(C(CCSC)O)=O)CC(NC(=O)CNC(=O)N(C)C)CC(F)C1 N1(C(=O)CCCN2CCOC2=O)CCC(c2ncc[nH]2)CC1 c1(C(=O)NC(CC#C)C)cc(CNC(c2c[nH]c(=N)o2)=O)cs1 Cc1cncc(C(=O)NCC2CCN2C(C2CC(=O)N(C3CC3)C2)=O)c1 C1(COC)(NC(c2sccc2C)=O)CCN(C(=O)CC2NC(=O)NC2=O)C1 C1(O)(CCNC(C(CC)=CC)=O)CCCN(C(=O)CC(O)c2ccccc2)C1 N1(C(c2cc(COC)no2)=O)CC2CC(NC(=O)C=CC(C)C)C1C2 Cc1noc(C)c1CSCC(=O)NCC1CCN(C(=O)CCSC(F)(F)F)C1 CCCCCCC(=O)NC1CCN1C(=O)C(=Cc1ccccc1)NC(=O)OC c1(OCC)cc(NC2CCSC3(C2)CC(C(=O)OC)C3)ccc1[N+](=O)[O-] Cc1ccc(F)c(C(N2CCC(F)C(NC(=O)CCOCC3CCCO3)C2)=O)c1 c1(C(=O)NCc2c(-n3cc(NC(C)=O)nn3)cccc2)cc2cccnn2c1 C(=O)(C(C)(C)S(C)(=O)=O)N(C(C)CNC(C1CC1C(F)(F)F)=O)C N1(C(C23C(CN(C(c4n(C)c(Cl)cn4)=O)C2)COC3)=O)CCCC(N=[N+]=[N-])CC1 N1(C(CCc2c(OC)cccc2)=O)CC2CCC(C1)N2c1ncc2c(n1)CCC2 N1(CC(N2CCC(OC)(CNC(c3c(C)csc3Cl)=O)C2)=O)CCC(=O)NC1=O c1(C(=O)NC(C#C)C)cc(CNC(C2(SCC)CCC2)=O)no1 C1(CN(C)CC2(O)CCCCC2)Cc2ccccc2O1 Cc1cccc(SCC(N2CCC(CNC(=O)CC3CC4(CC4)C3)C2)=O)c1 c1(C(N(C(CNC(C2(C)CC2(F)F)=O)C2CC2)C)=O)ccc(C2CCC2)nc1 C1(C(=O)OC)C(NC(=O)Cc2cccc(C)c2Cl)C2CCCC12 c1(C(=O)NC2CCCC(NC(C3CC4(CC4)CO3)=O)C2)cc(Cl)cc(F)c1F N1(C(CC2(C)CCN(C(C3CCC=CCC3)=O)C2)=O)CC(C(N)=O)C2(CC2)C1 C=C=CCCC(=O)N1CCC(CC=C)(C(=O)NCCCSC(F)F)C1 c1(COC)n[nH]c(=NCC(C)(C)NC(C23CCCC2C3(F)F)=O)s1 c1(C(N2C(C)CCC(NC(=O)C=C(Cl)Cl)C2)=O)cnc2ccncc2c1 C123CCC1CN(C2)C(=O)CN3.CCC(C)C=CC(=O)N(C)NC(C1CCCC1)=O C1(C(N(C2COCC2(C)C)C)=O)CN(C(=O)CCc2ccn(C)n2)CCO1 C(CC(=O)NOCC(N)=O)N(C(=O)NC1C(C(=O)OCC)C1(F)F)C Cc1ncnc(C(=O)NC(c2cn(C)nn2)C(=O)NCc2nnc(C)n2C)c1C CC1CCC(O)(C(=O)NC(C2CCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)C)CC1 C1(C(C(=O)NC(C(=O)N(C2CCC2(C)C)CC)C)O)CCCCC1 C1(C(=O)NC(c2ccccc2)C(=O)N(CC#C)CCF)CC=CCO1 c1(C(=O)NC2CCC(NC(=O)C(O)c3ccsc3)C2)nc(Cl)c(Cl)s1 O(P(=O)(CC1CCN(Cc2ccc(N)cc2)CC1)OCC)CC C1(F)(CNC(C2C(CC)N(C)CC2)=O)CCN(C(c2coc(COC)c2)=O)CC1 C1(CNC(c2nc(OC)oc2)=O)(CO)CC12CCN(C(=O)CCN(C)CC)CC2 C1(SC(=O)C(Cc2ccccc2)C(C)C)CCCCCCC1.n12nnnc1C2C C1(NC(c2nc(CC)sc2N)=O)CC2CC1CN(C(=O)CNCC(C)(C)C)C2 C1(C(=O)NC2CC(CNC(c3sccc3Br)=O)C2)OCC2CCCC1C2 c1(CC)cc(C(N2CC(NC(=O)COC3CC=CC3)C(C)C2)=O)cc(Cl)c1 c1(C(=O)NC(C)C(C)NC(c2ccc(O)c(N)n2)=O)ccc2nnn(C)c2c1 c1(C(N2CC(N(C(=O)C(F)C3CCC3)C)C(F)C2)=O)c(F)cc(F)cc1F CCCC(CC)CCC(=O)NCC1(O)CCCN(C(=O)Cn2ncn(C)c2=O)C1 N1(C(CSC)=O)CC2(CCC(CNC(C3CCN(CC(F)(F)F)C3)=O)O2)C1 CC1(C)C(NC(C2CC(=O)N2)=O)CCN1C(=O)C(C1CCCCCC1)O c1(CC(=O)NC2C(NC(C(CC)(C)OC)=O)COC2)cc(C)c(Br)c(C)c1 CCC(C)(C)C(C)CC(=O)NCCC1CCN(C(c2cccn2C)=O)C1 C1(NC(C2(C)COCCO2)=O)CC=C(C(=O)N2CCCCC23CC3)C1 C(=O)(C1=NNC(C(F)(F)F)C1)NC(C(C)NC(=O)CCn1cnnn1)(C)C c1(CNC(CC2(OC)CCC2)=O)cnn(C)c1C(=O)NC1CN(C(Cl)COC)C1 C12CN(CC1C(C)C)C2=O.c1(C(=O)N)ccn(C(C)C)c1C.c1(COC)ncco1 c1(ON2CCCN(Cc3ccccc3)CC2)cc2c(cc1SC1CC1)OCCO2 C1(CNC(C(=O)NC(C)C)=O)CCC(C(=O)NCCC2CSC2)C1 Cc1ccc(C=CC(N2CC3CC3(CNC(c3sccc3C#N)=O)C2)=O)o1 N1(CCCC(=O)OC)CCNC(=O)CC1(C)C N1(C(c2cnccc2Cl)=O)CCCCC1C1CCCN1C(=O)C1=COCCO1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CCN(C(C1CC(CC)C1)=O)C2 c1(C(=O)NC(CNC(CCC2CC(C)C2)=O)(C)CN(C)C)ccc(CCF)cc1 c1(OC)ccc(Cn2nc(-c3ccn(C)n3)nc2Cc2nncn2C(C)C)cc1 c1(C(N2CCC(COC)(NC(=O)CC(C)(C)COC)C2)=O)ccn2cncc2c1 CCC(O)(CC)c1cn(C2CCN(C(=O)CC3(CSC)CC3)C2)nn1 N(C1CC2(CN(C(C3(C#N)CC3)=O)C2)n2ccnc21)C(c1c(C)cncc1)=O N1(C(C(C)C2CNC2)=O)CCN(c2ccc(C(F)(F)F)cc2)CC1 N1(C(CCc2onc(C)n2)=O)CC(C(=O)NCC(C)(C)N=[N+]=[N-])CC(C)C1 C1(CNC(c2ccns2)=O)CCN(C(C2CCC(CN3CCOCC3)O2)=O)C1 Cc1ccc2c(c1)C(C(=O)NC(c1cccc(C(F)F)c1)CNC(=O)C1CC1)C2 N1(C(CN(C(c2ccncc2)=O)CC)=O)CCC=C(C(=O)NC)C1 N1(C(C(C(C)C)SCC)=O)CCCC(C)(NC(c2cc(C)ccc2F)=O)C1 c1(-c2ccc(C#N)o2)csc(=Nc2cccc(Cl)n2)n1CCc1cocn1 c1(C(=O)NC(CNC(c2cc(CC)on2)=O)CO)[nH]c(=N)ccc1Br C=CC(CCC)CC(=O)N1CCC(C(F)C(N2C3COCC2C3)=O)C1 C1(CNC(Cc2nc(C)sc2)=O)CC2CCC1N(C(=O)CCn1ccc(=N)[nH]1)C2 N1(C(C(CC(C)C)C)=O)CCC2CCCC(C1)N2C(=O)C(F)=CC1CC1 c1(C(=O)NCC2CN(C(C(CC)C)=O)CC23CCC3)cc(F)c(Cl)cc1Cl N1(C(c2ccsc2Cl)=O)CC(CO)C2(C1)CN(C(C13CCC1C3)=O)C2 C1(C2CCN(C(c3nccc(Cl)c3F)=O)CC2)(NC(COCC(=C)C)=O)CC1 Cc1[nH]c(C(=O)NC(C2CCCN(C(c3scnc3Cl)=O)C2)C)c(C)c1[N+](=O)[O-] c1(C(C(=O)NCC)N(CCOCC)CCNCC)scc(C)c1C.C1CC(F)(F)C1 CC1(C(N2CCC(C)(NC(c3ccc4nnnn4c3)=O)C2)=O)CCC2(CC1)CC2 Cc1oc(CNC(c2ccncn2)=O)nc1C(=O)NCC(C)(C)CN(C)C c1(CC(=O)NC2(C)CN(C(c3cc(Br)cc(F)c3F)=O)C2)cc(F)cc(C#N)c1 C(=O)(C(F)(F)CCNC(c1cn(C)nc1SC)=O)NC(COCC)C O=C(C(F)(F)C(O)C1CC1)NCc1n[nH]c(O)n1.C1(C)CCCCN1c1ncccn1 N1(c2ccc(S(=O)(=O)N(C)CC3CCOC3)cn2)CCC2(CCCCO2)CC1 C(=O)(CCCCCNC(C1CC(F)C(=O)N1)=O)NCC=CC(=O)OC C#CCCCS(=O)(=O)N1CCN(c2cc(C(F)(F)F)[nH]n2)CC1 O=C(C(O)CCc1ccccc1)N1CCC(CCNC(C2(O)CCOC2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1CCCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 Cc1ccc(C(c2ccccc2)NC(C2CCC2)C#N)cc1 C(=O)(CCCCCCNC(c1cnn2ccccc12)=O)NC(C#C)CC1CCC1 N1(CCNC(=O)NC)CCC(=O)N(CCC2CCCCC2C)C1=O c1(CC(=O)NC2CN(C(C=CC(=O)NC)=O)CC2C)ccc(NC(N)=O)cc1 c1(NC2CC(F)(CNCc3cc(C)cc(C)c3)C2)ncc2c(c1C#N)CCC2 c1(CC)c[nH]c2ccnc(N(CCN)CCO)c12.S(C)(=O)(=O)NC C=CC(C)(C)CC(=O)NCCn1cnc(C(=O)NC2(CC3CC3)CCCC2)c1 C1(C(=O)NCC(CO)NC(c2cc3n(n2)CCCO3)=O)CCC2(CCOCC2)O1 C1(NC(C=CCC)=O)CN(C(=O)CCNC(c2ccccc2Cl)=O)CC1C(F)F N1(C(C2N(CCC)CCC2)=O)CC(O)CCC1C(=O)Nc1cccc(CCF)c1 c1(OCC#C)ccc(C(=O)NC(c2ccccc2F)C(C)C)c(F)c1 N1(C(C2(C#C)CC2)=O)CCCN(C(=O)C(C)(Cl)Cl)CCC1 N1(CC(=O)N(CCCN2CCCC2)C)CC(NC(=O)C=CCBr)C2(CC2)C1 N(C(=NCCCc1ccc(OC)cc1)N1CCCC(C)(C#N)C1)C(COC)OC c1(NC(c2ccc(-c3cc(F)ccc3F)nn2)=O)nc2cc(F)ccc2s1 Cc1nc(O)ccc1C(=O)NC1CC=C(C(=O)NC2(CO)CCCCC2C)C1 C(CC1=CCN(C(=O)CCCNC(C)=O)CC1)NC(CNS(SC)(=O)=O)=O C(C(C)(C)CC1CN(C(C2(CCF)CCC2)=O)C1)NC(C1C(C(=O)OCC)C1)=O c1(OCC=CC(=O)NCC#CCNC(=O)C=CC2CC2)ccc(F)cc1 S(=O)(=O)(c1cccnc1)N(CC(=O)N(CCC)Cc1ccnc(Br)c1)C N1(C(C2SCCCS2)=O)CC2(CCN(C(C3(Cl)CC3)=O)CC2)C1 CC1CN(C(C2(C(=O)N(C)C)CC2)=O)CC1NC(=O)C=Cc1cccnc1 C1(C(C)NC(C23CCC2CC3)=O)CCN(C(=O)C(N2CCCC2)C2CC2)C1 N12CCC3CN(CC13)N(C(C)(C)C)C2=O.c1(SC)csc(N)n1.c1(CC)scnc1Cl c1(OC)cc(CN2CCN(Cc3ccc(OC(C)C)c(Br)c3)CC2)cc(Br)c1 CC(CC(F)(F)F)C(=O)N1CCOCCC1C(N1CCC(CC(N)=O)CC1)=O C(=O)(C(CC(F)F)NC(=O)CC1CC1)NCC(C#C)C(C)C C1(C#N)(C(N2CCC(CN(C)C(=O)C3CC3)C2)=O)CCCC1 N1(C(c2c(CNC(CC(=O)NC3CC3)=O)noc2)=O)CCC(O)C(F)(F)C1 c1(C(N(C2CCC(NC(Cc3ccn(CC)n3)=O)C2)C)=O)cc(F)ccc1N c1(C(=O)NCCOC(C)(C)CNC(=O)CC2CNC(=O)C2)nnn2c1CCCC2 N1(C(=O)OC(C)(C)C)CC2(CCC(SCCCN3CCOC3=O)OC2)C1 C1(C(N2C(C)(C(c3cc(Cl)nc(C4CC4)n3)=O)CCC2)C2CC2)CCOC(=O)CC1 CC(C)(C)C(=O)NC1(C2CCCO2)CN(CC(=O)Nc2ccsc2)C1 c1(NC(C(C)=CCOC)=O)ccc(NC(=O)CCOCC(F)(F)C(F)F)cc1C CC(C)CC(C(=O)N1CCN(C(=O)C=CC2CCCCC2)C(C2CC2)C1)N(C)C CCCC(CCC)=CC(=O)NC(CN(C)C)C(=O)NSCC(C)(C)C(=O)OC c1(CC)nnc2c(C(=O)NC(C3CCCCN3C(c3cnns3)=O)C)cccn12 N1(CC(=O)NC2CN(C(c3cnc(CC)s3)=O)CC(O)C2)CCCCCCC1=O c1(N2CCC(NC(C3C(C)CCC3)=O)C(F)C2)cc(C#N)nc(C2CC2)n1 c1(CC(=O)N(C(C)CC#N)C)ccc(O)cc1 N1(C(CCC=C(C)C)=O)CC(C)OC2(CCN(c3cc(CC4CC4)ncn3)C2)C1 c1(CNC(C(C)(C)C2CC2)=O)cnn2c1CN(C(C1C3CC3C3CC13)=O)CC2 C1(C(=O)NC(C(C)NC(C=C(C)C(C)(C)C)=O)(C)C)Cc2cc(C)ccc2S1 c1(NCC2CCC(C(N(C)C)=O)CC2)ccc2ccnc(Cl)c2c1 C1(NC(CCNC(C)=O)=O)CN(C(=O)CCc2cc[nH]n2)C2(CCOC2)C1 CN1CCN(C(=O)COc2cc(F)cc(Cl)c2)C(CNC(C2CCC3CC23)=O)C1 N1(C(c2cnc(CC)nc2O)=O)CC2CCN(C(=O)CN(C)C(=O)C3CC3)C(C2)C1 C(=O)(CS(=O)(=O)CCO)NC1CCN(C(c2c(OC)c(=O)cco2)=O)CC1OC c1(OC)cncc(C(=O)NCCC(O)CNC(=O)C(C(C)C)N2CCC2)c1 C1(C(N2CCC3CCC(NC(CCC)=O)C32)=O)CNC(=O)CC12CCC2 c1(C(N(C(C)C(=O)NCCCCCO)CCC)=O)cncc(CC)c1 C1(C(=O)NC2(C(=O)NCC(O)(CO)CO)CCN(C)C2)CCOCC1(C)C N1(C(CC2C(C)CCO2)=O)CCC(NC(=O)CC23CCC(CC2)C3)C(O)C1 C(=O)(N=c1[nH]nc(Br)s1)c1nc(NC(c2ccc(-n3c(C)ccn3)cc2)=O)sc1 O=C(C1=NN(CCO)C(=O)CC1)N1CC(NC(=O)C#CC2CC2)C2(CC2)C1 C(=O)(C=C1SCC(=O)N1C)N(C)CC1N(C(C2C(C)C(=O)C2)=O)CCC1 c1(OC)cccc(C(N2CCC(C)(NC(=O)CNC(c3cc(Cl)ccn3)=O)C2)=O)n1 c1(OC(C)C(=O)N2CC(C(C)NC(=O)CC(O)C3CC3)C2)ccccc1 C=CCCCCCC(=O)N1CCCC(CCNC(=O)CC2CCN(C)CC2)C1 c1(C(N(C(C)CCO)C(C)C)=O)cc(Oc2ccccc2)n(C)n1 CCC(C(=O)N(C)CCc1ncon1)N(C)C(C1CCOC1)=O c1(C(=O)NC(C2CC(NC(C3(C)CCNC3=O)=O)C2)C)ccc2nccn2n1 C1(NC(=O)Nc2cccc(Cl)c2C(=O)NC2CC2)C(F)(F)C12CCOCC2 CC1(C)CCC(C(=O)NCCCN(C(c2ccc(C(N)=O)cn2)=O)C2CC2)O1 c1(C(C)(C)C)ccc(Br)c(C(=O)NC2CC2CNC(=O)CC2C=CCC2)c1 C1(O)(CNC(COC)=O)CCN(C(=O)C=Cc2csc(Br)c2)C1 c1(C(=O)NC2CCN(C(C3CCC(C)(C)CO3)=O)C23CC3)nc[nH]c2nccc1-2 C1(O)(CCNC(c2ncc(C)nc2)=O)CCCN(C(C2CC(F)C2)=O)C1 C1(NC(CC(CC)CC)=O)CCC2(CC1)CN(C(=O)Cc1cnn(C)c1C)C2 N1(C(CC(C)N(C)C)=O)CC2CC(O)C1C2NC(=O)CCS(N)(=O)=O C1(C(=O)Nc2c(C)ccc(F)c2)CC2CCC(C1)N2C(c1csnc1Cl)=O C1(C(N2CC(c3ccccc3)(NC(C(C)=C(C)C)=O)C2)=O)CC12CCOC(C)C2 c1(OCC)ccccc1CCC(=O)NCCC(C)N(C(=O)CC(C)OC)CC N1(C(=O)C(C2CC2)C2CC2)CCC(NC(C2(c3cccnc3Cl)CC2)=O)C(O)C1 C(C(C)(C)C#CC(=O)N1CCC(CC(N)=O)C1)NC(CC(C=C)(C)O)=O C(=O)(C(C)C1=CCCC1)NC(CC)CNC(c1ncoc1C1CCC1)=O C1(CC(=O)NCCN2CCCC2=O)(NC(C2C(C)(C)C2Cl)=O)CCCCC1 C1(NC(c2c(C(=O)OC)c[nH]n2)=O)CCCCC1NC(=O)CC(C)(C)C C1(O)(CN(C(=O)CCCCCn2cnnn2)C)CCCN(C(=O)C2=NOCC2)C1 c1(C(=O)NC2(CN(C(=O)CN(C3CCC3)C)C)CC2)cnn2ccc(Cl)c(F)c12 Cc1cn2ccnc(C(=O)NCC3COCC3NC(C3(N(C)C)CC3)=O)c2n1 c1(N2CCCC(CNC(C3CCCCC34CCC4)=O)C2)ccc([N+](=O)[O-])cc1Br CCCC(C(=O)N1CCC1c1cn(-c2ccccc2C(=O)O)nn1)OC N1(C(c2c(CC)nn[nH]2)=O)CCCC(O)(CCNC(=O)C=CBr)C1 N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCOCC(CNC(=O)CC2(C3CC3)CC2)C1 CC(C)CC(C)C(=O)N1CC(C)(NC(c2cnc(N3CCOCC3)cn2)=O)C1 C(=O)(C1SCCc2ccccc21)NCC1N(C(c2[nH]c3ncn(C)c3c2)=O)CC1 C(=O)(C(CNC(c1nscc1C)=O)C(C)(C)C)NCCNC(=O)NCC C1(C=O)CC2CC(=O)C1O2.C(=O)(C(CNC1CC1)N(C)C)N(C1CN(C(C)C)C1)C N1(C(c2n(C)ncc2)=O)C(C(=O)NCC#CC2CC2)CCC1C1CC1 C1(C#N)(C(N(C(CNC(C2CC23CCC3)=O)C2CC2)C)=O)CC1(C)C CCCC(CC(C)C)C(=O)N1CCC2CN(C(=O)CCCC(C)(C)C)CC12 CN1CCCC(O)(CCNC(=O)NCc2ccnc(OC3CC3)c2)C1 c1(C(C)(C)C)ncn(C)c1C(N1CCC(F)(C(=O)NCC2CCO2)C1)=O N1(C(C2C3CC4C(C3)C24)=O)CC2CCCC1C2CO.CC1(N)CC(n2ccnn2)C1 CCC(C)CC(=O)N(C1CCN(C(C2CCC(N(C)C)CC2)=O)C1)CC N1(C(C)C)CCC(N2CCC(NC(=O)C(=O)NC3CC3)C2C)C1=O C1(C(=O)NC(C(C)(C)C)C(=O)NC2CC3CCC(C2)O3)CC(=O)CC12CCC2 Cc1sc(=O)n(CC(N2CCC2CNC(C23CCC2CC3)=O)=O)c1C N1(C(c2c(CC)c[nH]c2)=O)CCCC(C(C)(O)CNC(=O)Cc2c[nH]nc2O)C1 N1(C(Cn2nc(C)oc2=O)=O)CCCN(C(=O)Cc2scnc2C)C(C)C1 C1(CC(=O)NCC)CCCN(C(C2CNC(=O)C2)=O)C1 c1(C(=O)NC2CCCC2NC(C2CC(F)(F)C2)=O)cc2c([nH]1)CCCC2 c1(NC(CN(C(=O)CCCN(C)C)CC#C)=O)c(C)noc1C C1(NC(c2nc[nH]n2)=O)CC2CCC(C1)N2C(=O)CN1CSCCSC1 CS(C)(=O)=NC(=O)C(=O)N1CCC(C2(NC(c3cnc4ccccn34)=O)CC2)C1 C1(CNC(C2CCCC2(F)F)=O)CN(C(c2cscn2)=O)CC12CC2 CCC(CC(=O)NCC12CC1CN(C(c1cnc(S)nc1)=O)C2)C(F)F c1(NC(C2(NC)CC2(C)C)=O)ccc(OCc2ccccc2)c(Cl)c1 c1(C(=O)NC2CCC3CCN(C(CCCCOC)=O)C32)cncc(P(C)(C)=O)c1 CC1OC2CCC1(NC(=O)C=CC1CCN(C(=O)OC(C)(C)C)CC1)C2 C1(CNC(=O)C(N2CCCCC2)C2CCCC2)CCCOCC1 N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(CCNC(=O)CSc2cn[nH]c2)CC1 c1(C(=O)OC)ccc(CC(=O)NC2(C)CCN(C(=O)C=C(C)C)C2)cn1 c1(OC)nc(C)ccc1C(=O)NCCC1(NC(=O)CC2CC2)CCC1 N1(C(=O)CN2CCCC2)C(C(N2CC(F)C2)=O)CCC1C.c12cnn(c1)C2.N1CCC1 C1(CNC(c2c[nH]c(=NC)s2)=O)CCCCN(C(C2CNC(=O)CC2C)=O)C1 c1(CNC(C2(CC(=O)OC)CC2)=O)nocc1C(=O)NC1CC(N(C)C)C1 C(C)(C)(C(CO)CO)N(c1cccnc1)C1C(C)CC1 c1(OC)ccc(NC(=O)C(N2CCOC(c3ccc(Cl)cc3F)C2)C)c(Cl)c1Cl c1(C(N(C(C2CCC(C)(C)C2)C(=O)NCCCSC)C)C)nc2ccccc2[nH]1 c1nc2c(N3CCC(OCCO)CC3)[nH]c(=NCc3cccc4nsnc34)nc2s1 C(CN=c1nc2sccc2c(CN2CCCC(N3CCCCC3)C2)[nH]1)OCCC C1(C(=O)NCCC(CC)(C)NC(=O)C(C)CC2CCC2)CC2CCC1CC2 C(=O)(C(C)(C)CC(C)C)N(C)CC1CCN(C(CSc2ccc(C)cc2)=O)CC1 Cc1[nH]nc(Cl)c1C(N1CCC(CNC(=O)C=CSCc2ccco2)CC1)=O C1(C(=O)NC(CCc2onc(CC)n2)=O)CC12CCOC(C)C2.C12CN(C1)N2C N1(C(C(CC#C)C)=O)CC(NC(c2cnc(SC)nc2O)=O)CCC1C C1(C(=O)NCC(CN(C(C2C(CCOC)C2)=O)C)C)Cc2c[nH]cc2S1(=O)=O c1(OCC(N2CC(C(=O)Nc3cccnc3)C(O)C2)=O)cccc(C(F)F)c1Cl C1(CNC(C2(C#C)CN(C(C3CCCOC3)=O)C2)=O)CCC2(CC2)CO1 C(CC(C)C)(C(=O)NC1CCN(C(c2cccc(OC)n2)=O)C1(C)C)OC C12(NC(CC(CCC)O)=O)CCCC1N(C(c1cccc3[nH]ccc13)=O)CC2 Cc1cc(CC(=O)NC(CNC(c2cncn2-c2ccccc2)=O)CO)n[nH]1 N1(C(C2(CSC)CCC2)=O)CCC(CO)(CNC(C2CC(S(C)(=O)=O)C2)=O)CC1 N1(C(C2CN(C(C)=O)C2)=O)CCC(C)(CNC(=O)CCCC2CCC2)C1 C(=O)(C1=CCC2CCC1N2C(C1CCC(C)(C)C1)=O)N1CC(C)SCC1 CCC1=NOC(CNC(C2(NC(c3cc(C)co3)=O)CC(CO)C2)=O)C1 N1(C(C(C)n2ccnc2)=O)CCC(C(C)C(=O)C(=O)CN2CCC3CC23)CC1 C1(C(=O)NCC2(CO)CC(C)C2)CCN(C(=O)C2CC(=O)C2)O1 C1(C2CC2)(C(N2C(C(=O)NC)COCC2)=O)CN(C(=O)CC2CCCC(O)C2)C1 N1(C(=O)CC2(O)CCC2)CC2CCC2(CNC(=O)CCOC2CC2)C1 N1(Cc2c(C#N)scc2)CC2CC1CN2C(c1snc(Cl)c1Cl)=O c1(C(N2CC(NC(c3cnc(CC)s3)=O)(CO)C2)=O)ccc(CC)c(OC)c1 Cn1ccc(C=CC(=O)NCC2CCCCN2C(c2cnn(CCO)c2)=O)c1 C1(=CC(N2CCC(NC(Cc3cnc(C)o3)=O)C(C)C2)=O)CC2CCC(C1)N2C C(=O)(CS(=O)CCC(F)(F)F)NCC1(CNC(C=Cc2ncn(C)c2)=O)CCC1 C1(CNC(c2n(CC)nnn2)C2CCCO2)CCC2(CCCC2)CC1 Cc1cccc(C(=O)NC(CC(N)=O)C(=O)NCc2n[nH]cc2C2CC2)c1N C1(CC(=O)N(CC(CNC(C(C)OCC)=O)(C)C)C)CC(=O)NC1=O c1(C(=O)NC(CC(C)NC(C(C)=C2CCCC2)=O)C)cc2oc(Cl)cc2[nH]1 C1(C(N2CCC(OCC#C)C2)=O)CC=CC(NC(c2ccnc(OC)c2)=O)C1 CC1CN(C(c2ccc(F)cc2F)=O)CC(CCNC(c2csc(CO)n2)=O)O1 C1(N(C)C(c2cnc(Cl)s2)=O)CN(C(=O)CN2CCCC2C(N)=O)CC12CC2 C(=O)(C(O)CCCNC(=O)C(C)=CC1CC1)N(CC)CC c1(C(N2C(CNC(=O)C(=O)Nc3ncc[nH]3)CCC2)=O)cccc(Cl)c1C(F)F C1(NC(c2cn(C)nn2)=O)COCCN(C(C2(c3cccs3)CCOCC2)=O)C1 C(CCC(C)(F)F)NC(C(N1CCC(n2cc(CSC)nn2)C1)=O)=O CC1(CCO)CCN(C(c2cccc(CC(F)(F)F)c2)=O)C1.c12cc(ncn1)N2 C(=O)(CCCN(C)N=O)NC1CN(C(c2cc(OCC)n[nH]2)=O)CC1(C)C N1(C(C=CCN(C)CC)=O)CCC(NC(c2ncn(C)n2)=O)C(CO)C1 C=CCC(C(=O)N1CC(C)(C)C1)NC(c1c[nH]ccc1=O)=O C(=O)(C(C)(F)C(C)(C)F)NC1CC(CC(=O)N(CC(O)CF)CC)C1 N1(C(=O)OCC)CSCC1C(=O)NCCC1CCN(C(=O)C=CCF)C1 C1(C(N2CC(O)(CNC(c3ccc(C)s3)=O)C2)=O)CCC2(C1)CC2(F)F C1(C(N(CCC(N)=O)CC)=O)CCN(C(=O)CCc2cncnc2)C(C)(C)C1 C(C)(CO)(C(=O)NCCC(C)NC(C1(CO)CC1(F)F)=O)NC(C)=O N1(C(c2c(C)cno2)=O)CCC(C)(CNC(c2cscc2C#N)=O)C1 C(=O)(NN1CCc2ccc(F)cc21)c1c(NC(=O)OC(C)(C)C)cc(Cl)cc1 C12(C(=O)NCC(CN(C(CC3(OC)CCCCC3)=O)C)C)CC1COC2(C)C C1(NC(CCCN(C(=O)C#CC2CCCC2)C)=O)CCn2ncnc2C1 C(=O)(C1COc2ccc(Cl)cc21)NC1C2(CN(C(C3C(=C)CC3)=O)C2)SCC1 N1(Cc2ccc(NCCN(c3ccc(OCC)cc3)C)cc2)CC(C)OC(C)C1 CCC(CC)C(C)C(=O)N1CCCC(CC(N2CCC(O)(CC)C2)=O)CC1 c1(C(=O)NC(C)Cc2cccnc2)cc2n(n1)CCCN(Cc1ccsc1)C2 C1(CC(=O)NCCCN(C(c2cn(CCN(C)C)nn2)=O)CC)CCCC(C)C1 N1(C(CC2(C)CC2)=O)CCC(CNC(c2cnn(C3CC3(F)F)c2)=O)C12CC2 Cn1cc(C(N2CC(CNC(=O)CSCC3CCCO3)C2)=O)c(O)n1 N1(C(c2c(CC)nc[nH]2)=O)CC(CNC(c2cccc(C)c2)=O)CC12CCC2 N1(C(C(CNC(CCSCCC)=O)N(C)C)=O)C2CCC1CN(C)C2 CCC(=O)CCC(=O)N1CCC(CCNC(=O)CC2(OCC)CC2)CC1 C1(C(=O)NC(C(=O)OCCC)(C)C)CN(C(C2CC(C)C2)=O)CC1CCC N1(C(C2(SC)CC2)=O)CCCC(CCNC(=O)COCC2CCCO2)CC1 C(=O)(CCCC(=O)NCCC(C)(C)CNC(=O)CC1(C)CC1F)NCC c1(C(C(=O)OCC)NC(=O)C(O)CC2CCCCC2)c(F)cccc1Br Cc1cc2[nH]c(C(N3CCC(C(=O)NCc4cccc(C#N)c4)C3)=O)cc2o1 N1(C(C2C(COC)CC2)=O)CC(O)CC1CNC(=O)CCSCC(N)=O CC(CCC(=O)NC1CC(NC(=O)CCCc2ccccc2)C1)Nc1nccs1 C(=O)(CCS(=O)(=O)NC)N1CCC(N(C(C2C(C(=O)OC)C2)=O)CCO)CC1 c1(C(=O)NCC(C)N(C(C(C=C)c2ccccc2)=O)CC)cc(C)c(C)c(C)c1 C(=O)(C(CCC1CC1)NC(c1cc(Cl)n(C)n1)=O)NC(c1nc(C)[nH]n1)C C(=O)(CCC(C(C)C)NC(c1nn(C)cc1C)=O)NCCC(C)N(CCC)C C1(C(N(CC(C)NC(=O)Cc2ccsc2)CC)=O)CC12CCCCCC2 c1(C(=O)NCC2CN(C(C)=O)CC2C)c(C)nn(C)c1Br C(=O)(CC(C)CNC(C12CC(CN1C(C1(CF)CC1)=O)C2)=O)OCC C12(CNC(c3ccc(CCC)[nH]3)=O)CCC(CC1)N(C(c1n[nH]c(C)c1C)=O)C2 N1(C(C(C)OCCCC)=O)CCC(C(=O)NCc2cc(C)co2)C1C c1(CC(=O)NCCN(C)C(C2CC2(C)C)=O)ccc2c(c1)CCCO2 c1(C(=O)NCC(CNC(c2cnn(CC)c2C)=O)OC)cnc(C(F)F)c(C)c1 C1(C(=O)NCC(C)CNC(=O)CSc2cccs2)(COCC)CCC1 C1(C(=O)NCC2(C)CNC(=O)O2)CN(C(c2cc[nH]c2)=O)CC1C1CC1 CCCC(C)(C)CC(=O)Nc1cc(N2CCC(C(=O)OC)C2)nc(C(F)(F)F)n1 N1(C(CSC(C)C)=O)CCCC1(C(=O)NCC1C2CCCOC12)C(C)C C1(CC=C)(NC(=O)CC2CC=CCC2)CCN(C(c2ccc(N)cn2)=O)CC1 C1(NC(c2oc(CC)c(C)c2)=O)CC2CC1N(C(C1(CSC)CCC1)=O)C2 c1(C(=O)NC2CCN(C(c3c(C)nc(CO)s3)=O)CC2)ccc2c[nH]nc2c1 Cn1ccc2cc(C(=O)NCC(Cl)NC(=O)CCc3ccc(F)cc3)cnc12 N12CCC(F)(CC1)CNC2=O.c1(COc2n(C)ncc2CO)cc2scnc2[nH]1 N1(C(C=C(COC)C)=O)CC(C)(C)CCC1CNC(c1ccc(C)cn1)=O C1(CCNC(C(C)c2ccsc2)=O)COCCN1C(=O)CCc1ccccc1Cl c1(C(N(C(C(N2CCN(CC)CC2C)=O)CC(F)F)C)=O)ccc2cc[nH]c2c1 CC(=O)CCCC(=O)N1CCC(CNC(c2ccc(C3CC3)cc2C)=O)CC1C N1(C(c2c(C)nc(C3CC3)o2)=O)CC2CC(N(C)C(c3cnn(C)n3)=O)C1C2 Cc1ccc(F)cc1C(=O)NCC1CN(C(C2CC(C(C)C)C2(C)C)=O)CC1C CC(C)C(C)(O)C(=O)N1CCCC(C)(NC(c2coc(C(N)=O)c2)=O)C1 c1(CC(N2CC(C)(C)C(NC(=O)COC3CCCC3)C2)=O)ccc2ncnn2c1 C(C(CC)CC(C)C)NC(C(=O)NCCN(C(COCCCC)=O)C)=O c1(CC)cc(C(=O)NC(CNC(c2c[nH]c(=N)s2)=O)CC)cc(F)c1 N1(C(C(C=C)OC)=O)CCCCC(CNC(=O)C(CC)n2ccnc2)C1 n1(CCC)cncc1CNC(C1CCOC1CNC(=O)CSc1nc[nH]n1)=O CC(O)(Cc1ccccc1)C(=O)NC(CNC(c1coc(C(F)F)n1)=O)CO c1(C(=O)NCCOC2CN(C(C3(C)CCCS3)=O)C2)cc2c(o1)CCCC2 C1(CC)C(NC(=O)C(=O)NCC(F)(F)F)CCCN1C(c1ccnnc1O)=O C(=O)(CCCN=[N+]=[N-])N1CC(NC(CNc2c(NC(C)=O)cccc2)=O)C(C)C1 C1(N(C(c2n(CC)ncn2)=O)C)CN(C(c2cc(C(C)(F)F)n[nH]2)=O)CC1O N#Cc1ccc(Cl)c(CN2CCC(F)(F)C(NC(=O)Cc3ccc(O)nc3)C2)c1 C1(NC(c2c(O)ccc(OC)c2)=O)COC2C(NC(=O)CC(C)CF)COC12 c1(C(=O)NC23CC(CNC(c4ncc(C)cc4F)=O)(C2)C3)cc2cc[nH]c2cn1 c1(C(=O)NC(CNC(C2CCSCC2)=O)C2CC2)ccn2cncc2c1 C(CC(C)C(=O)NC1CC(CNC(c2ccc(N(C)C)nn2)=O)C1)OC c1(N(C)CCC2CCCN2C)nc(=NCCCCC#N)[nH]c2c1SCC2 N1(C(C(CCCC)ON=C(C)C)=O)CC2CCC1C(NC(=O)CC1C=CCC1)C2 c1(CNC(C=C(C)CNC(c2cnnc(O)c2)=O)=O)cnc(C)cc1C CN1CCN(c2nccc(CC(=O)O)c2Br)CC1CO N1CC2(C1)CN(C(=O)C(F)CC1CCOC1)C2.C1(C(=O)C=C)CCOCC1 CC(C)CC(CNC(=O)C1=CCCCC1C)C(=O)NC12CCCC1OCC2 C#Cc1ccc(Cl)c(C(N2CC3CC(C2)N(C(=O)C(C)CCCC)C3)=O)c1 C1(NC(=O)COC(F)(F)F)CCCCN(C(=O)CCC2CCCCCC2)CC1 Cc1cccc(C)c1CNC(c1nnnn1C)(c1nnnn1CCCF)C CCC(CNC(C1CSCCN1C(=O)CN1CCCCC1)=O)C(C)(F)F C(CNC(C1CCOC(C)(C)C1)=O)(CC(F)(F)F)NC(c1c(CC)onc1C)=O N#Cc1c(C(=O)Nc2ccc(-c3cccnc3)cn2)sc2c1CCC2 N1(C(Cc2ccn(C)n2)=O)CCCC(F)(CNC(c2cccc(CCO)c2)=O)C1 CCC(CCCC(=O)NCCC(C)(C)CO)NC(C1CCS1(=O)=O)=O C1(C(=O)NCC2CCCN(C(=O)CCCCC3CC3)C2)CC12CCSCC2 Cc1cccc(CNc2ncc(-c3cnn(C4CCOC4)c3)s2)c1 Cc1cccnc1CC(=O)Nc1ccc(CSc2ncc(-c3ccccc3)s2)s1 C1(CC)CCCC1C(=O)NCC(CO)NC(=O)C(C)(C)C1CC1 N1(C(CSCCC)=O)CCCCC(NC(=O)CCCCNC(=O)OC)C1 N1(CC(N2C(C)CC(CNC(C=C(C)C)=O)C2)=O)CCCc2sccc2C1=O C1(CNC(C2C(C)C2C)=O)CC2COCC2N1C(c1cn(C2COC2)nn1)=O Cc1cc(C)n(C(C)CNC(c2cnn(CCNC(C3COC(=O)N3)=O)c2)=O)n1 C#CCCC(C(=O)NC(Cc1ccco1)CO)NC(C1CCCC(CF)C1)=O C1(N(C(c2c(C)n(C(C)C)nc2)=O)C)CCN(C(=O)CCCC2CC2)CC12CC2 c1(CC)nn(C)c(CC)c1C(N1CCC(CO)(CNC(c2cc(C)no2)=O)C1)=O c1(OC)ccc(C(=O)NCCC2CN(C(c3sc(C)cc3OC)=O)C2)cc1 C1(NC(=O)CC(C(F)F)NC(=O)Cn2ccnn2)CCOC2(CCC2)C1 C#Cc1ccc(C(=O)NCC2(F)CCN(C(=O)Cc3ccsc3)C2)cc1 C1(CC=C)(NC(C2CC3C=CC2C3)=O)CCCN(C(=O)C=Cc2sccc2C)C1 c1(C(N2CCN(C(CCOC)=O)C(CF)C2)=O)ccc(S(=O)(=O)N(C)CC)cc1 C(C(C)(C)CC(=O)N1CC2(CCC2)CC1C(N1CCCOC(C)C1)=O)OC C1(O)(CNC(C(CC)NC(=O)CC2CC(C)C2)=O)CCCOC1 n1(CCC)ncc(-c2csc(C(=O)NCCc3ccoc3)n2)c1CC N1(C(c2cncc(CC)c2)=O)CC2(CCCN(C(c3cc(Br)co3)=O)C2)C1 Cc1ccc2c(c1)C(C(=O)NCCN(C(c1ccc(F)c(Cl)c1F)=O)C(C)C)C2 CCC(CNC(c1cc2cnccc2[nH]1)=O)N=c1ccc([N+](=O)[O-])c(O)[nH]1 CC1CCCN(C(C2CN(C3COC3)C2)=O)C1CNC(=O)CC1CCCCCC1 N1(C(C2(CC=C)COC2)=O)CCC2CCN(C(c3ncc(N)cc3C)=O)C2C1 c1(CC2(C(c3nnnn3C)NC(=O)OC)CC(CC)C2)ncc(OC)cn1 N1(C(CCc2cc(OC)cc(=O)o2)=O)C2CCC1CN(C(=O)CNS(C)(=O)=O)C2 c1(C2CCN(C(=O)OC(C)(C)C)C2)ccc(F)cc1.c12n[nH]cc1oc(=O)s2 c1(C(N2C(C#C)CC2)C(=O)NCCC2(C)CC2)ccc(S(N)(=O)=O)o1 c1(SC(C)(C)C)ncncc1CNC1CN(C(=O)CCC2CCCO2)C1 N1(C(C2COC3COCC23)=O)CCCN(C(=O)C(F)(F)C(F)F)CC1 CCC(C)(CC)C(=O)N1CCOC(C)(CNC(=O)COc2ccccc2Cl)C1 N1(C(c2c(CC)csc2)=O)CCC2CCCC12CNC(c1cnccn1)=O c1(C(=O)NC(C(CO)NC(CC2ON=C(C)C2)=O)C)c(C)c2cnccn2c1C Cc1ccc(NCC(N2CC(c3ccccc3)(NC(=O)C(C)(Cl)Cl)C2)=O)cc1 c1(C(N2C(C(C)NC(C3(C=C)CCCCC3)=O)CCC2)=O)ccc2c(c1)COC2 c1(OC)ccncc1C(N1CCOC(C(C)NC(=O)CC2(OC)CCC2)C1)=O c1(OC)cc(CC(=O)NCC(C)NC(=O)C(CC#N)c2ccccn2)cc(Cl)c1 C(=O)(CCCc1cnn[nH]1)NC(C1CCCN1C(=O)CCOC1COC1)C C1(CCC)CCC(O)(C(=O)NCC2(F)CCCN(C(C3(O)CCC3)=O)C2)CC1 C(C)(C(C(=O)NCc1ccccn1)C(C)C)NC(Cc1ccc(C)s1)=O C1(C)(CC)CCC(C(=O)NC2CC(C)(CNC(c3nc(C(C)(C)C)no3)=O)C2)O1 CC1(C)C2CCC1(C)C2C(=O)NCCC1CC(NC(C2CCC(C)(F)CC2)=O)C1 CCC(CC)CC(=O)NCC(C1(O)CCN(C(=O)CCN2CCCC2=O)CC1)C Cn1cc(C(N2CC3C(NC(C4CC45CCCC5)=O)C3C2)=O)c(C(F)F)n1 c1(CN(CCNC)CCF)nc(CC)cc(C#N)n1.C(=O)(C(=O)NC(C)(C)C)N c1(NC)nc(C)ccc1C(=O)N(CCCOCCNC(=O)CC(C)F)C N1(C(c2n(CC)ccn2)=O)CCC(C)(C)C(NC(=O)COCCOCCOC)C1 c1(CC(=O)NCC(C)NC(C2CCN(C3CC3)CC2)=O)c[nH]c2c(F)cccc12 CCC(C)C(O)C(C)C(=O)NCC1CCC(C)CN1C(c1ccon1)=O c1(OCCOC)ccc(C(=O)NC(C)CNC(C2CS(=O)(=O)C2)=O)cc1 C(=O)(CS(=O)C(F)(F)F)NCC1(OC)CCN(C(C2(F)CC2C)=O)CC1 C(C(C)(C)C(=O)Nc1cn(CCF)nc1C)NC(c1nc(CCC)oc1)=O C1(NC(C(C)(C)N2CCCC2)=O)CN(C(=O)CCc2cnoc2)C2CC12 c1(C(=O)NC2C(CNC(CNC(C3C(C)C3)=O)=O)C2)c(Cl)cc(Cl)c2ncccc12 N1(CCNC(C2(F)CCC2)=O)CCCN(C(=O)Cc2ccccn2)CC1 C(=O)(C1=CC2C=CC1C2)NC(CCOC)C(=O)NCC1(C(C)C)CC1 c1(SC)cccc(C(=O)NC2CCCN(C(C3CCCN3C)=O)C2)c1 Cc1cc(C)c(C(=O)NC(C)(C)CCNC(=O)CC2CCCOCC2)[nH]1 c1(C(=O)NCC(CCc2ccc(C)cc2)OC)cccc(C(C)NC(CC)=O)c1 CN1CCN(C(C2CCOC(=O)CC2)=O)C(CNC(=O)CCNC(N)=O)C1 N1(C(C(C(C)O)C)=O)CCCCC12CC(NC(c1cc3ccccc3o1)=O)C2 c1(C(CNC(=O)CCc2cnoc2)NC(C=CC=CCC)=O)cc(F)cc(Cl)c1 CCCCC(CC)C(=O)N1CCC(N(C(=O)Cn2ccnn2)CCC)CC1 c1(C(N(C2CN(C(C(CC)N3CCCC3=O)=O)C2)C)=O)nn(C)c(Cl)c1Cl c1(SC)ccc(F)cc1.C12CCN(C1)C(=O)CN(CC1CC1)C2 N1(CC(=O)N(CCNC(CCOCC)=O)C(C)C)CCc2ccccc21 c1(CCC(=O)NC2(CCCNC(C(CC)=CC)=O)CC2)ccc2[nH]ccc2c1 CCC(C)(COC)C(=O)N1CCC(C)(CNC(=O)CCn2cnccc2=O)C1 C1(C(=O)NC2CC(OC)C2)(C(=O)NC(C)CC2(O)CCCC2)CCCC1 C(=O)(C1=CC2(CCN(C(C3CC3(C)C(F)F)=O)C2)C1)NC(C#C)C1CC1 C1(O)(C(C)NC(CCSC(C)C)=O)CCN(C(c2cc[nH]c2)=O)C1 CCCC(CNC(c1ccncn1)=O)C(=O)N(C1(C)CC1)C c1(C(=O)NCC(C(C)C)NC(c2ncccc2Cl)=O)nccc2c1CNC2=O C(=O)(C(C)C(C)(F)F)NCC(C)CNC(=O)CN(CC(=O)NC(C)C)C C1(C#N)(c2n(-c3c(C)cccc3C)nc(C(F)F)n2)CC12CCCC2 CCCCC(C(=O)NC1CN(C(=O)CS(C)(=O)=O)CC1CO)ON=C(C)C CC(CC(F)(F)F)C(=O)NC1(C)CCN(C(c2n[nH]c3c2CCSC3)=O)C1 c1(C(=O)NCCCC2(NC(c3ccc(C4CC4)cc3)=O)CC2)occ2c1CCC2 N#Cc1cc(Cl)c(C(N2CC(O)(CCNC(=O)CCN3CCC(O)CC3)C2)=O)s1 C(=O)(C1CC(=O)c2c(F)cccc21)N1C2CN(C(C3C(=O)OCC3)=O)C(CC2)C1 C1(CC)CCC(C(N2CCCCC2CN(C(=O)CNS(N)(=O)=O)C)=O)CC1 c1(CCC)nc(C(=O)NCCNC(=O)C(=O)OC(C)=O)c(C)o1.c1(N)ccc(OC)cc1 c1(-c2cn(CC(C)OC)nn2)c(NC(C2(C)CC2Br)=O)cnn1C c1(N2CCC(C=C)C2)nc(N2CCC(C3CC3)C2)c2c(n1)CCS2 Cc1csc(C(=O)NC2CC(N(C(c3sccc3OC(F)F)=O)C3CC3)C2)c1 C1(C(N2CCC(CCOC)C2)=O)(CC)CCCN1C(=O)Cc1cncn1C Cc1cccn2c(-n3cc(C4CCN(C(c5ncoc5Br)=O)C4)nn3)cnc12 N1(C(C(C)OCC#C)=O)CCC(C2(CNC(=O)C=CCCC)CCOCC2)CC1 Cc1cc(C(=O)NC(C)(C)COC(C)(C)C)sc1-c1ccccc1Cl N(C(=NCCCCCS(C)(=O)=O)NCc1ccc2[nH]ccc2c1)C(CC)C Fc1ccc2cnc(NC3CN(Cc4ncc(Br)cc4F)CC3(F)F)nc2c1 c1(OC)ccc2c(c1)CCC1C2OCCN1C(=O)Cc1ccccn1 C(CCCCNC(=O)C(F)=CCCF)N(C(=O)CCn1ccnc1)C C1(CNC(c2c(C)nsc2)=O)CCN(C(C23CCC2C3)=O)CC1(F)F C(N=c1nc2c(c[nH]1)C1CCC2C1)c1cc(C(=O)OC)c(Br)cc1 N1(C(CCC#CC)=O)CCCC(C2CCN(C(=O)C(F)(F)CC)CC2)CC1 C12CCCCC1NC(=O)NC2.Cn1ccnc1-c1cc(NC(=O)C(F)(F)F)on1 C1(C(=O)NCCCSCC)CCN(C(=O)C=CCOC)C12CC2 C(=O)(C1CCc2ccccc21)NC(C(=O)N(CCCCC=C)C)(C)C C1(NC(CNC(CCC2C(C)(C)C2)=O)=O)(CO)CC(F)(F)C1 C1(C(=O)NC)CCN(C(=O)CN(C(C2CC3(CC3)C2)=O)C(C)C)C1C c1(C(=O)NCCCC(C)NC(C2C=CCC2)=O)ccc2c(c1)nc(O)n2C1CC1 C12(NC(c3c(Cl)cn(CC)n3)=O)CCN(C(c3ccc(N)c(F)c3)=O)CC1C2 C1(C(=O)N)CC2CCC1C21CC1.C1(COCC)CCN(C(c2cc(CO)[nH]n2)=O)CC1 O=C(C1CCCc2nc[nH]c21)NC1CN(C(c2cnc3c(c2)COC3)=O)CC1O C1(CCCC)CC(C(=O)N2CCC(c3cn(Cc4ccc(Cl)s4)nn3)C2)=NO1 N1(C(CCOC(C)C)=O)CC2CCC(C1)N2C1CCN(C(C2CCC2C)=O)CC1 c1(C(N2CCC(N(C(C3(C)CCN(C)CC3)=O)C)C2)=O)csc2cccnc12 C1(CNC(C2CC(N(C)C)C2)=O)CN(C(C2(C(N)=O)CC2)C)CCO1 C1(C)(C(=O)NC2CCC(NC(c3ccc(C(C)C)o3)=O)CC2)CCN(C)C1=O CCC(CC)(C(=O)NC1CC(CNC(=O)Cc2nc(C)sc2C)C1)C(C)C N1(C(c2cccc(C(=O)NC)c2)=O)CCC2CCN(C(C3CCC(=O)N3)=O)C2C1 N1(C(C(C(COC)C)C)=O)CCC(C2(O)CN(C(=O)CCCCSC)C2)CC1 c1(-n2cc(CNC(c3cn(CC(CC)C)nn3)C)nn2)ccccc1OC C1(N(C)Cc2onc(CCC)n2)CCN(C(C2(C3CC3)CCC2)=O)CC1 N1(C(C(=Cc2cnc[nH]2)C)=O)C(CNC(c2cc(Br)n[nH]2)=O)CC2CC12 C=CCCCCCC(=O)NCC1C(O)C(O)CN1C(c1cc(CC)sn1)=O c1(C(N(C)CC2(O)CN(C(C(CC)SC)=O)C2)=O)cccc(CF)c1 c1(CNC(c2ccc(C(C)=O)[nH]2)=O)ccc(Cl)cc1F C1(C(=O)NC2CC(CCNC(c3ccsc3C(F)(F)F)=O)C2)C2CC3C(C2=O)C13 Cc1cn2c(n1)C(C(=O)N1CC(CNC(C3CC(F)(F)C3)=O)C3(CC3)C1)CCC2 c1(CNC(C2CC(NCc3ccc(Cl)nc3)C2)=O)ccnc(Br)c1 C1(CN(C(COCC(=O)NC)=O)C)CCN(C(C2(NC(N)=O)CC2)=O)CC1 N1(C(C(CC)C#N)=O)Cc2nccn2CC(C(=O)NCc2ccc(C)c(C)c2)C1 c1(C(=O)NC(C(C)O)C(=O)NC(C)(C)C)nccc(I)c1C(C)(C)C O=C1CCC(C(=O)NC(C(N2CCCC2CCCO)=O)C2(O)CC2)C1 Cc1cc(C)nc(Sc2nc(C(C)C)c(C)s2)n1.c12ocnc1CNC2=O c1(C(=O)NCC(C(C)C)NC(c2ccc(CO)cn2)=O)cncc(N)c1 N1(C(c2nc(CC)oc2)=O)CCC(C(N2CCC(C)(N(C)C)C2)=O)(CCOC)C1 N1(C(c2c(NC)cccc2)=O)CCCCC(C(=O)NCCCN2CCC2)C1 c1(C(N2CC(CCO)(NC(C3CCC(=O)C3)=O)C2)=O)ccc(F)cc1F CCC(C)C(=O)C(=O)N1CCC(C)C1C(=O)NOCCc1ccccc1 C1(C(C)C(=O)N(C)C2CC2)CCN(C(=O)C=Cc2ccco2)C1.C12CN(C1)C2 Cc1cnn(C(C)C(N2CCC(n3cc(C(=O)Nc4cn[nH]c4)nn3)C2)=O)c1 c1(SCC)ccnc(NCC2(NC(=O)C(F)(F)C3CCOCC3)CCC2)n1 C1(CC=C)(C(=O)NC(C2CCCN2C(c2cnc(C(C)C)[nH]2)=O)C)CC=CC1 c1(C(=O)NC2CC(NC(=O)C=Cc3cscn3)C(O)C2)cc2c([nH]1)CCCC2 C(C)(CS(=O)(=O)CC)n1c(CC(CCC)C)nc(-c2ccccn2)n1 C=CCC(CNC(c1cc(CO)n(C)n1)=O)C(=O)N1CC(CO)C1(C)C Cc1cccc(Br)c1-n1cc(C(C2CCN3CCCC23)=O)nn1.C1(C)CCOCC1 c1(C(N2C(C)(C(=O)Nc3ncc(Br)cc3Cl)CC2)=O)ncc2ccccn12 c1(C(C(=O)NCCC(=O)NC)NC(=O)CC2C(=O)NN=C2C)c(C)cccc1Br C1(C(=O)NC(C2CCN(C(=O)C(c3cnn(C)c3)=O)CC2)C)CCOC2(CCC2)C1 N1(C(C(CC)NC=O)=O)CCC(C(=O)Nc2ccc(Cl)nc2C(F)(F)F)C(O)C1 C1(CC(=O)NC2CC(C(=O)OC)CC2O)C(=O)NCCN1C(=O)CC(C)N(C)C CC#CCCCC(=O)N1CCCC1(C(=O)NC(C1CCOC1)CO)CCOC CC1CNc2c(C(=O)NCCNC(=O)CNC(=O)C3CC3)cccc2C1 CC1(C(=O)NC2CN3CCC2CC3)CC(F)(F)CN1C(=O)CCCC(F)(F)F CC1(N)C=C(C(=O)NC2CCC(NC(C3CCCC4(CCC4)O3)=O)CC2)C=C1F C12(C(=O)NC3C(NC(C=C4CCN(C)CC4)=O)CCOC3)CC(C)(CCO1)C2 N1(C(c2cnc(C3CC3)o2)=O)CCC2CC2(C(=O)N(C2CCC2)CCN(C)C)CC1 N1(C(CN2CCC(C)CC2)=O)CCC(C)N(C(=O)Cc2nn(C)cc2Cl)CC1 C=C(C)CCC(=O)N(C)CC1CN(C(c2sc(COC)nc2C)=O)CCO1 c1(N(CC(F)(F)Cl)C(C)C)nc2ccccc2nc1NCCCc1cc[nH]n1 N(C(=NCC1CCNC(=O)C1)NCC1COCCO1)CC1(S(C)=O)CC1 C1(NC(=O)CNC(c2ccccc2Br)=O)CC2CN(C(=O)C=C3CC3)CC2C1 C1(NC(c2cc(C)oc2C)=O)C(CN=c2nc(C(C)C)[nH]s2)CCC12CCC2 C(CCC(=O)NC1(CCNC(=O)Cn2cnnn2)CCC1)OC N1(CC(=O)NC(CCCNC(c2c(OC)ccs2)=O)(C)C)CCS(=O)(=O)CC1 Cn1nc2c(c1C(=O)NCC1(NC(c3cccc(O)c3Cl)=O)CC1)CCC2 N1(C(c2cc(C)cc(C)c2)=O)CCC2CN(C(c3c(Br)cnn3C)=O)CCC12 CC(C)CC(C)(C)C(=O)NCC1CC(O)(CNC(c2cc(Cl)ccc2F)=O)C1 c1(NC(c2c(C)nsc2N)=O)ccc(OC(F)F)cc1F S(=O)(=O)(c1ccc2c(ccn2C)c1)N1CC(NC(C2C(C)C2)=O)C(F)CC1 c1(C(=O)NCCn2cc(CC3(O)CCSC3)nn2)cc(O)ncc1F N1(C(C2CC(CC)(CC)C2)=O)CCC(F)(C(=O)N(C2CC2)Cc2ccoc2C)C1 CCCC(C(=O)NCCC1(O)CN(C(=O)C=C(C)C)C1)S(N)(=O)=O C(=O)(CC1=NNC(=O)C1)NC(CCCNC(Cc1c(SCC)cccc1)=O)C N1(C(c2c(Cl)ccc(C)c2)=O)CCN(C(=O)C=Cc2ccncn2)CC12CCC2 Cc1cn2cc(SCC(N3CCCCC3c3cc(O)nc(S)n3)=O)nc2s1 C1(CNC(c2cnc(SC)s2)=O)CC(=O)N(c2ccc(-c3ccc(Cl)s3)cc2)C1 c1(C2C(C(=O)NCCCN(C(CC)COC)C)CCO2)cncc(Br)c1 c1(C(N2CCC(C)C(N3CCC(C)C3)CC2)=O)cc2nccn2c(O)n1 C(C(CC)(CC)C(=O)NCC1CNC(=O)CO1)NC(C(C=C)O)=O CCC(CC(=O)NCCN(C(c1ccccc1)=O)CC)C1CCC1 C(=O)(C(=O)C(C)(C)C)NCC(C1CCCC1)NC(C(CSC)O)=O N1(C(C2C(=C)C2)=O)CCCN(C(c2cscc2Cl)=O)CC1C C1(CNC(CCC(=C)C)=O)CC2(CO1)CN(C(C1CCCC(C)(C)CC1)=O)C2 C(=O)(C1=CCCCO1)NC1C(OC)CN(C(c2cccc(Br)c2C)=O)C1 Cc1cnc(C(=O)NCC2CC(C(=O)NC3(C(F)(F)F)CC3)C2)c(F)c1 c1(C(=O)NC23CC2CN(C(=O)CCCC2CCOCC2)C3)cccc2c1OCO2 c1(C(=O)NCCCOCCNC(C=C(CC)CC)=O)ccc(=O)n2c1CCCC2 C1(CC(=O)NCCCC(C)(C)NC(c2ccn(C3CC3)n2)=O)CC2CCC1CC2 c1(CNC(=O)OC)ccc(C(=O)NC(C)CC(C)NC(=O)CCCC(C)C)cc1 C1(NC(C(C)OC)=O)CN(C(c2ccccc2C(F)(F)F)=O)CCC12CCC2 C1(C(=O)NC(C2CN(C(c3coc(C(F)F)n3)=O)C2)C)CN(C)CCO1 N1(CC)CCN(C(C2(CCNC(=O)C(C)CC(=O)OC)CCCC2)=O)CC1C CCCC(C(=O)NCCOC1CCN(C(=O)C(CC)OC)CC1)S(N)(=O)=O c1(NC(C23C(CN(C(c4ccncc4Br)=O)C2)C3)=O)cccnc1F C1(CC(=O)N(C)CCNC(C2CC3CCC(C2)O3)=O)CCc2ccccc2C1 N1(C(c2[nH]cc(CN(C)C)c2)=O)C2CCC1C(NC(=O)Cn1nccn1)C2 O=C(CCCCCF)N1CCN(C2CCN(C(C3(N(C)C)CC3)=O)C2)CC1 N1(C(CNC(C2(C)CC2)=O)=O)CCOC2(CCN(C(=O)Cc3nc[nH]n3)CC2)C1 c1(N2C(C(C)C)CN(Cc3ccc(C(=O)O)s3)CC2)ncnc2cnccc12 C(CCCCC(=O)NC1CCC1NC(c1n[nH]c(C)c1Cl)=O)OC N1(C(CSCC#C)=O)CCC(C)(CNC(=O)C(C)Oc2cccc(F)c2)CC1 c1(C(=O)NCCCN(C(=O)CC2CCC(=O)NC2=O)CC)ccc(O)c(F)c1 CC1(C)CC(CNC(=O)C(CCF)NC(c2ccccc2)=O)CO1 C(CC(C)C(=O)NCc1cc(C)c(C(=O)N(CCF)CC)o1)=CC C1(CCNC(c2ccoc2Cl)=O)CC2CCC(C1)N2C(=O)CN1CCCNC1=O C(=O)(CCCCCNC(=O)CC(C)=C(C)C)NC(C(CCC)O)CO C(=O)(CC(C)C(F)(F)F)NCCCC1OCCN(C(c2nc(C)nc(O)c2)=O)C1 c1(C(N2C3CN(C(C45CC(C)C4C5)=O)C(CC3)C2)=O)ccc2ccccc2n1 C1(C(N2CCC(N(C(C(CSC)C)=O)CCO)CC2)=O)CCC=CCC1 c1(C(N2C(C)CC(CNC(c3ccc(C#N)s3)=O)CC2)=O)cccc2[nH]ncc12 CC(C)C(O)C(C)(C)C(=O)N1CCOCC(C(=O)NC(c2n[nH]c(CO)n2)C)C1 N1(C(C(CCC)C(C)C)=O)CCCC2(CCCN2C(=O)C(F)C2CCC2)C1 C1(CCC(=O)NC2(C)CN(C(=O)COCc3nccs3)C2)CCCC(O)C1 c1(C(N2CC(C(C(=O)NC(C#C)CC3CCCC3)OC)C2)=O)cscc1Cl C(CN=c1[nH]cnc(NCc2ccc(Br)c(C)c2)c1C)(c1ccsc1)OC c1(C(=O)OC)cc(C(=O)NCC2(NC(C3CC3Cl)=O)CCC2)cc(O)c1 C1(CCNC(CCS(C)=O)=O)CN(C(=O)CCN2CCC(O)CC2)CCCO1 CC(CCNC(=O)C(CNC(=O)C#CC(C)(C)O)CC1CCCC1)C(C)(C)C c1(CS)cccc(NC(C2CC(C(N3CC(n4cc(CC)nn4)C3)=O)C2)=O)c1 N1(CC)CC(C(=O)N(C2CCN(C(c3cc(C)co3)=O)C2)CC)CCC1=O N1(C(c2c(SCO)n(-c3ccc(Cl)cc3F)nn2)=O)CCCOC(CN=c2nc[nH]s2)C1 C1(O)(CCNC(CN(C)C(C2CC2F)=O)=O)CN(C(C2CCCCC2)=O)C1 Cc1cc(C)n(CC(=O)N(CCCNC(=O)C(C)C(C)c2ccccc2F)C)n1 C1(OC)(OC)CCC1C(=O)NC(C)(C)CN(C)C(C12COCC1C2)=O C12(C(=O)NCC3C(C(N(C4CC(OC)C4)C)=O)OCC3)CCC(C1)OC2C c1(C(=O)NCCC2(CNC(CC=CC=C)=O)CC2)cccc(Br)c1C C1(CCNC(C=C(CC)C)=O)CN(C(C23CCC(C2)C3)=O)CC(C)O1 Cc1cn(C)nc1C(=O)NC1CCC(C)(CNC(c2cnc(S)nc2)=O)C1 N1(C(Cn2c(C(C)C)nnn2)=O)CC2CCC1CN2Cc1ccc(Cl)cn1 C1(C)(CNC(C2CCC(C)C2)=O)CCN(C(=O)CC(F)(F)F)CC1 c1(N(C(c2cn(C)nc2)=O)CCNC2C3COCC23)ccc(Br)c2ccccc12 C1(N(C(C(F)(F)C2(OC)CCC2)=O)C)CCCC(N(C(=O)Cc2cnc[nH]2)C)C1 c1(C(N2CC(C(=O)NCC(F)(F)F)C2)=O)ncsc1NC c1(C(=O)NC2(CNC(c3ncn(CC)c3)=O)CCC2)c(Br)ccc(C)c1N C1(C(=O)NC)CC2(CCN(C(=O)CN3CCNC3=O)CC2)C1 N1(C(C(CC)N(C)C)=O)CCC2CN(C(c3cccc(C#N)c3)=O)C2C1 C1(NC(C=CCC)=O)CCN(C(c2cnn(-c3nccs3)c2)=O)C(C)C1 N1(C(C(CC=C)NC(c2cccc(C)c2C)=O)=O)CC(C)OC(C)(C)C1C N(C(=NCCF)NCC1OCC1(C)C)CC1(OC)CCCCC1 N1(C(C)C)C(=O)COCC1C(N1CCC(CN(C(=O)C(=O)NC2CC2)C)C1)=O c1(CC)ccc(C(N2CCC(NC(c3cc(N)cc(O)n3)=O)C2C)=O)cc1Cl c1(C(N(C(C)Cc2ccccc2)CC)=O)cncc2c(F)cccc12 c1(NC2CCCO2)cc(N(C)CC2CN(C(COC(C)C)=O)C2)nc(C(C)C)n1 C1(CNC(C(C)OC(c2c(F)ccc(C)c2F)=O)=O)COc2ccccc2O1 C1(C(N2CCC(NC(COCc3n(C)ccn3)=O)C2)=O)CC(C)(C)CC(C)(C)C1 c1(C(N2CC3C(CNC(=O)CC4CCSCC4)(C3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(c2c(C)cccn2)=O)CCN(C(=O)CC2CCC3(CC2)COC3)C2CCC12 S(=O)(=O)(c1ccc(=NCCCCCC#N)[nH]c1)NCc1c(SC)ccc(Br)c1 C1(C(N(CCN(C)C)CCO)=O)CN(C(=O)Cc2nn(C)cc2Br)CCC1O c1(NC(C(=O)NC(c2ncon2)C)=O)cccc(S(=O)(=O)CF)c1 CCC(CC)CCCC(=O)N(CC(C)CNC(c1occ2c1CCC2)=O)C N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CCC(C(F)(F)F)CC1C c1(NC(C)=O)cnc(O)c(C(=O)NC2CC(CNC(=O)C=C3CCC(C)C3)C2)c1 c1(N(C)CCC2CCCO2)ccc(Br)c(S(=O)(=O)NCC2CCc3ccccc32)n1 C(=O)(CC(C)(C)C(F)F)N(CC(C(=O)NC(C(C)SC)C)C)C N1(C(C)=O)CCCC1C(=O)NC1CC(C)(C(=O)N(C)CC2CN(C)C2)C1 N1(c2cc(NCCCN3CCCC(C)C3)nc(C)n2)CCCC2(CCSCC2)C1 N1(C(CC(=O)OCC)=O)CCSCC1C(=O)NCCC1CCN(C)CC1 C1(NC(NCCOC)=NCC2CCn3ccnc3C2)CCCC2(CN(C3CC3)C2)O1 c1(OC)ccc(Br)c(C(=O)NCC2CCC2NC(=O)C(C)N(C)C)c1F c1(C(=O)NC2CC(CO)N(C(=O)C=CBr)C2)cccn2cncc12 C1(NC(CC2(N(C(CCC(=O)NCC)=O)C)CC2)=O)CCCC(C)CC1 C1(CC)CN(C(c2c(C)noc2C(C)C)=O)CCN1C(=O)C(n1cc(Cl)cn1)C CC(C)(C)CCC(=O)NCCC1CN(C(C2(C)CCOC2)=O)CCO1 c1(N(CCOC)C(=O)OC(C)(C)C)ccc(OC)cc1.C(C)(C(F)(F)F)NC(=O)N c1(OC)c(C)cc(N2CCN(CC(c3cc(C)sc3C)=O)CC2)cc1C C(=O)(CC(O)CNC(C12CC(C#N)(C1)C2)=O)N(CCNC(C(C)C)=O)C C1(SC)C2CCC(C2)N1C(=O)CCn1cc(-c2cnn3c2NCC3)nn1 C1(C(=O)NC2(CNC(C(CC=C)NC(C)=O)=O)CCCC2)CS(=O)(=O)CC12CC2 CC(C)C(C(C)N(C)C)OC(=O)CC1CCC2(CC2)C1 N1(C(Cc2c(C)ncs2)=O)CCC(C)(C)CC1C(=O)NCC1CCOC1(C)C CCCC(C(O)C(=O)NCC1(C(C)(C)OC)CC1)NC(c1cccc(C)c1F)=O N1(C(Cc2cnc(C)s2)=O)CCC(O)(CN(C)C(C2CC(C)(C)O2)=O)CC1 C1(n2cc(NC(C(C)C)CO)nn2)CCCN(C(=O)CSC(=N)N)C1 C1(C)(C(=O)NCC2CCN(C)CC2)CN(C(C2CCOC2(C)C)=O)C(C)(C)C1 CC1=C(C(=O)NC2CCC3CC2CN3C(c2ccc(C(N)=O)[nH]2)=O)CCCO1 c1(OC)cccc(S(=O)(=O)N2CCC(C(=O)N=c3[nH]oc(C)c3Br)(F)C2)c1 c1(C(=O)NC2(CNC(C3C(C)CC(=O)N3)=O)CCC2)cncn(C)c1=O c1(OCCCC)ccc(C(=O)NCC2(O)CCN(C(=O)CCCN(C)C)C2)cc1 Cc1nn(C)cc1C(O)C(=O)NCCC1(O)CN(C(=O)CCc2cn(C)nn2)C1 c1(CCC)cc(C(N2CC(CNC(=O)C(C)(C)SC)CC2C)=O)nn1C c1(C(=O)NCC(C)(C)NC(CCc2cnc(C)s2)=O)cnn(C2CCCC2)c1C c1(C(=O)NC(CC)CN(C)C(C2CC2(C)C)=O)ccnn1C(c1ccccc1)C C(CC(C(=O)NCC1(C(C)(C)OC)CC1)NC(C1CC=CC(O)C1)=O)OC c1(CN(C(C(C)NC(C(C)c2cccs2)=O)=O)C)nc(C2CC2)no1 c1(C(=O)NCC(CN(C(=O)C(c2ccccc2Cl)(C)C)C)O)cccc(O)c1F N1(C(C(CC)COC)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(C(C)C)C1 CC1=NOC2(C1)CC(C(=O)NC(C)(C)CNC(=O)CCc1ccc(F)c(F)c1)C2 C(CC(=O)NCCCCN(C)C(c1ccccc1CO)=O)(C(F)(F)F)OC CC(C)C(CNC(=O)Cc1cncn1C)C(=O)NCC(C)(C)O c1(COC(C2CC3CC(NC(=O)OC(C)(C)C)C3C2)=O)cccc2ccccc12.OC c1(CC)noc(C)c1C(=O)NCC1(NC(=O)CC2CC23CC3)CCOC1 C1(C(N(CC(C)(C)CNC(=O)Cc2cc(C3CC3)no2)C)=O)CCC=CCC1 Cc1nc2c(cc1C(=O)NC(C)C(C)NC(=O)CCNC(=O)CO)c(C)nn2C C(=O)(C1=CCCSC1)NCCCc1cn(-c2c(COC)cccc2)nn1 CCCC(C)(CCC)C(=O)N1CC2(NC(c3ccn(CCO)c3C)=O)CC1C2 C(=O)(CCS(=O)(=O)NC1CC1)N(CC(CC)NC(=O)CSc1ccccc1)C c1(C(N2C(CCNC(C3C(C)(Br)C3)=O)CSCC2)=O)coc(S(N)(=O)=O)c1 O=C(C1CCCn2cnnc21)NCC1(F)CN(C(=O)Cc2cnn(C(F)F)c2)C1 CCC(C)(CNC(=O)CCCCCNC(=O)Cc1cccnc1F)C(N)=O c1(C(=O)NC2C(C(=O)NCCc3cc(C(=O)OCC)no3)C2)scc(C)c1Cl C1(O)(CC(N2CCC(N(C(=O)Cn3ncc(Br)n3)CC)C2)=O)CCOCC1 C1(CNC2CCN(C(C)C)CC2)CC(C)(C)CN1C(=O)CC(C)n1ccnc1 c1(C(=O)NCC2(F)CCCN(C(C(C)(C)OC)=O)C2)cccc2occc12 N1(CC(c2c(C)cccc2)C)C(=O)CN(CCCCCc2ccc(F)cc2)C1=O N1(CCN(C)C(C2(O)CC2(C)C)=O)CCN(C(C2CCCCC2O)=O)CC1 C1(NC(C(CC)OC)=O)CC2C1CCN2C(c1cc(F)ccc1O)=O N1(C(c2ccc(N(C)C)cn2)=O)CCN(C(=O)C2=C(Cl)CCC2)C2CC12 c1(N(C)C)ccc(C2C(C(=O)NC3CCCC3NC(=O)CO)C2)cc1 C1(CCNC(C(C)NC(N)=O)=O)CSCCN1C(c1ccncc1F)=O C1(C(=O)NC2C(NC(c3cc(C(F)(F)F)ns3)=O)CC2)CC2CCC1CC2 C1(NC(c2ccc(-c3cccs3)cc2)=O)CN(C(C2(O)CC2)=O)CCC1F C(=O)(CCCCF)NC(CC(C)NC(CCCOC)=O)C Cc1ncc(CC(N2CCC(CNC(=O)CC3COC(=O)N3)CC2)=O)c(O)n1 c1(OC)noc(C)c1C(=O)O.C(C#CC)C(N1CCC1)=O C(=O)(CC(O)c1ccccc1)NCCC1(CNC(=O)C(C2(O)CCCC2)O)CC1 CC#CCCCC(=O)NC(C)CCCNC(C1(C#N)CC1(C)C)=O C(=O)(C(C)CCO)NCC1N(C(CN(CCC)C(=O)OC(C)(C)C)=O)CC1 c1(CN2CCC(CNC(c3nnn(CC)c3C)=O)C2)ccc(C)c(C)c1 C1(NC(CC2C(C)(C)C2)=O)CC2CC1CC2C(=O)NC1CCSC1 c1(COC)ccccc1NC(C12CC(CNC(=O)C(CC)SC)(C1)C2)=O c1(C(=O)NC(C2(O)CN(c3snc(CC)n3)C2)C)cnc(O)cc1OC C1(CN(C(c2[nH]c(C)nc2C)=O)CC)CCN(C(C2CS(=O)(=O)C2)=O)CC1 c1(-n2cc(C3(C(=O)NC4(Cl)CC4)CCN(C(C)=O)C3)nn2)cccc(Cl)c1F C1(C(=O)NCCCCOC)(NC(c2ccc(C)c(C)c2)=O)Cc2ccccc2C1 Cc1c(CN2CCCC2)cccc1Br.C12CC3CCC1(C3)NC(=O)N2 C1(NC(C2(F)C(C)C2)=O)CCCC2CN(C(c3cc(O)nc(Cl)c3)=O)CC12 c1(C(=O)NC2CC(CNC(Cc3nc(CC)sc3)=O)C2)cccc2c1COCC2 N1(C(CC2(C)CCCC2)=O)CCC2(CCC2NC(c2cscc2Cl)=O)CC1 C(CNC(C1CC1c1ccco1)=O)(C(=O)NCCc1ccoc1)N(C)C c1(C(=O)NCCCN(C(c2[nH]ccc2C2CC2)=O)CC)cc2nc(F)ccc2o1 C(=O)(C1=NOC2COCC12)N1CCC(C)C(CC(=O)NCCS(C)(=O)=O)C1 C12(CNC(c3c(C)cc[nH]3)=O)CC(NC(C3CC4CCC3C4)=O)(C1)C(C)(C)O2 C1(N(C(c2cnn(CCO)c2)C(=O)NC2CCOCC2)CC)CCCCC1C C(C)(C(=O)NCC(O)C(=O)NCCc1cnc(C)o1)(C(C)C)OC N1(C(C(=O)NC(CC)C)=O)CCC2(CCC(=O)NC2)C1 C(=O)(C1=C(C)CCCC1)NC1(CC=C)CCN(C(=O)CCc2cncc(O)c2)C1 c1(C(=O)NC(CC(C)C)CO)cc2c(-c3cnn4ccccc34)cccc2s1 N#Cc1c[nH]c(CNC(=O)NCCCC2CCCO2)c1 C1(NC(=O)Cc2cnoc2)CCCN(C(=O)Cc2ccsc2Br)C1 N1(C(CC(CNC(CC2(C)CC2)=O)C2CCC2)=O)CCC(C2CCC2)C1 C(C(CC(C)C)C(=O)N1CCCC2(C1)N=N2)NC(c1cc(CC=CC)no1)=O c1(C2(C(N(CC(CN(C(=O)CSC(F)(F)F)C)O)C)=O)CCC2)ccccc1F Cc1cc(C=CC(=O)NC2CCCC(CNC(C3CC=CCO3)=O)C2)c[nH]c1=N N1(C(c2cc(C)n(C)n2)=O)CCN(C(=O)CC2(O)CCCCC2)C(CC(N)=O)C1 c1(NC(C)=O)ccc(C)c(C(=O)NC23CC(C2)N(C(C2CCC(C#N)C2)=O)C3)c1 C1(C(=O)NCC(CC(C)C)NC(CCOC)=O)CCCC2CCCCC12 N1(C(CCn2c(C)nc(C)n2)=O)CCOC2(CCC(NC(=O)C(F)F)CC2)C1 O(N(C)C(=O)C(CNC(C1C2CCC(F)C12)=O)CC(C)C)CC(=O)OC N(C(=NC1CCC1)NC1CCOCC1)CC(O)COc1ccc(C2CC2)cn1 c12cc(ccc1Cl)C(=O)N2.N1(CC)CCC(C(N)=O)C(O)C1 C1(NC(c2ncc(C)nc2)=O)CC2CN(C(=O)C(C)N3CCC3)CC12 c1(OC)ccc(F)cc1C(=O)NC1CC(CNC(=O)CCCN=[N+]=[N-])C1 CC1CN(C(c2occc2CNC(c2ccc(Cl)cc2)=O)=O)CCC1CO C(=O)(CC(C)(C)CN(C)C)N(C1(CNC(=O)CC23CCCC2C3)CC1)C N1(C(C(C2CCN(C(Cn3ccc(C)n3)=O)C2)F)=O)CCNC(=O)C1 Cc1c(C(=O)NCC2CC(C)(C)Oc3ccccc32)ccc2c1CCC2 c1(C(=O)NCCCC2N(C(C(CC)=CC)=O)CCCC2)ccc(P(C)(C)=O)cn1 C#Cc1ccc(C(=O)NC(CNC(c2cc(OCC)no2)=O)C(C)CC)cc1C c1(OC)cccc(C)c1NC(C)CC(C)O c1(C(=O)NCCOC2CCN(C(C34CC(CF)(CO3)C4)=O)C2)nccc(Cl)c1F N1(C(c2nccc(COC)c2)=O)CCN(Cc2cc(Cl)c(Cl)cc2F)CC12CC2 N1(C(Cc2cccc(OC)n2)=O)CCCC(CO)(NC(C2CC2C(C)O)=O)C1 CC(C)(C)C1CC(=O)N1.C1(C(CC2CC2)=O)CCSC1 c1(NC2CC(CNC(C(CC)C)=O)C2)ncc(Cl)c(O)n1 c1(N(CC(=O)NCCC)C)nc2cc[nH]c2c(=NC(CC)c2nc(C)cs2)[nH]1 Cn1nnc(C(=O)NC2CCCN(C(c3ccnn3CCF)=O)C2)c1C(F)F N1(C(C2CCC(N(C)C)C2)=O)CC2CCN(C(c3coc(O)n3)=O)CC12 Cc1nc2ccc(C(=O)Nc3csc(-c4cnn(CCCN(C)C)c4)n3)cc2[nH]1 c1(OC)ncc(F)cc1C(=O)NCC1CC1CNC(=O)C1=COCCO1 c1(C(N2CCC(C)C(NC(=O)Cc3cncnc3O)C2)=O)noc2c1COCC2 C(=O)(C(CNC(C1CCC(C)(C)OC1)=O)CC(C)C)NCC(CC=C)(C)CO C1(NC(c2cnc3cccnn23)=O)CN(C(c2csnn2)=O)CC2(CC2)C1 C#CCC(O)C(=O)N(C1CCCCC1)CC1CCCN(C(=O)C2=COCC2)C1 c1(C(N2CCC(CS(C)(=O)=O)C2)=O)c[nH]c(NC(=O)OC(C)(C)C)c1 C1(C(C)(C)C)CCN(N2CCN(S(=O)(=O)Cc3ccccn3)CC2)C1 c1(C(N2CCC(C)(C(=O)OCC)CC2)C(=O)NCC)ccc([N+](=O)[O-])cc1.N(C)CC c1(C(=O)NCCOC(C(=O)N(C(C(=O)NC)CC)C)C)cncnc1C CCC(C)CC(C)C(=O)NCc1ccccc1CNC(c1cnn[nH]1)=O c1(CC(N2CC3C(NC(C(C)=C4CC4)=O)C(C3)C2)=O)cncc2ccccc12 c1(C(N(C(C)C)Cc2cccs2)=O)nc(C(F)(F)F)ccc1F C(CC(C(=O)NC1(C(=O)NC(c2ncccc2C)C)CC(O)C1)OC)OC N1(C(c2n(C)cc(C#N)c2)=O)CCC2C(C1)CN2C(C1CCCOCC1)=O CC(O)C(C)(C)CNC(=O)C(c1ccccc1)NC(C1CC1(F)Cl)=O Cc1ccc(C(=O)NCCCCC(=O)NC2(CO)COC2)cc1 n1(CC(N2C(C)C(NC(C3CC34CC(O)C4)=O)CCC2)=O)cc2ncccc2n1 Cc1cc(C(N2CCOC(C(N3CCS(=O)(=O)CC3)=O)C2)=O)c(F)cc1Br c1(NC(C2CCCCN2C)C)cc(N2CCOC(CN(C)C)C2)ncn1 C12(CNC(c3occ(C)c3)=O)CCC(NC(=O)Cc3nonc3C)(CC1)CO2 Cc1sc(N)c(C(N2CCC(C(C)NC(=O)CCOC(C)C)C2)=O)c1C c1(C(=O)NC(C(C)NC(c2cc(CC)n(C)n2)=O)(C)C)cccc2c1ncn2C C(N=c1[nH]c(=NCc2ccncn2)[nH]c2cccnc12)c1c(C)scc1 c1(C(N2CC(C)C(NC(=O)CNC=O)CC2)=O)ccc2c(c1)C=CS2(=O)=O c1(C(=O)NC2CN(C(c3cncc(C)c3)=O)CC2C#N)c(Br)ccc(F)c1F c1(C(=O)NCC(C)N(C)C(C2(F)CC=CC2)=O)c(N)ccc2nccnc12 N1(Cc2cnn(C)c2CNC(C2(O)CCCC2(C)C)=O)CC2C3C=CC(C3)C2C1 N#Cc1ccccc1CN1CC(CN(C2CCCCS2)Cc2ccco2)CC1=O c1(CC(=O)NCC2C=CC(CNC(C3C(C)C3)=O)C2)cccc(Br)c1F N1(C(c2ccc(Cl)nc2)=O)CCC(N=c2[nH]nc(C3CC3)s2)C2(CCC2)C1 c1(C(N2CC(=C(CNC(CCCCCC)=O)F)C2)=O)cc2c(=O)[nH]ccn2n1 N1(C(Cc2c(C)noc2C)=O)CC2CCOCC2(NC(c2coc(Cl)n2)=O)C1 CCC(CCO)C(C)NC(=O)N(CCO)Cc1ccco1 C(=O)(C1=NNC(=O)CC1)NC(C1CCCCN1C(C1CCC(=O)N1C)=O)C c1(NCC(=O)NC(CC)CNC(C2(CC(F)(F)F)CC2)=O)cncc(Br)c1 n1(CC(=O)Nc2ccc(OC(F)(F)C(F)F)nc2)cc2ccccc2n1 C(=O)(C1=C(Cl)CCC1)NCC(C)(C1CC1)NC(c1c(C)nn(CCO)c1)=O C1(C(=O)NCC(CNC(c2ccc(C(=O)OC)cc2)=O)C)CN(C)CCN1C C1(C)(C(=O)NCCC(CNC(c2cc(CCCCC)[nH]n2)=O)O)CCC(=O)N1 c1(C(=O)NCC2(CNC(C3(C(N)=O)CC3)=O)CCC2)cc2ccccn2n1 C1(NC(=O)Cn2nnc(=O)[nH]2)CCCCCC1NC(c1ccoc1C(F)(F)F)=O C1(NC(c2cc(OCC)no2)=O)CCN(C(=O)C(CO)N(C)C)CC(C)(C)C1 CC12CC(NC(C3CCCOC3)=O)(C1)C1(CN(C(=O)C(F)(F)C(F)F)C1)O2 C(=O)(C1=NOC(C)C1C)NC(C1CCN(C(C(C)c2ccsc2)=O)C1)(C)C N1(C(c2c(C)ncs2)=O)CCN(C(c2ccncn2)=O)C(C2CCCC2)C1 c1(C(=O)NC2C(NC(C(C(CC)O)(C)C)=O)CCC2)ccnc2c1ncn2C N1(C(Cc2cnc(C)[nH]2)=O)CC2(CCCC2NC(=O)C=Cc2cn[nH]c2)C1 C1(CC(N2CCC(COC)(CNC(=O)CC(C)CF)C2)=O)CCC(C)(C)CC1 C=CCCC(CCC=C)(c1nnnn1CCC#N)NCc1cc(C(C)(C)C)no1 C(CS(=O)c1ccccc1F)NC(=O)Cc1cc(Cl)ccc1Cl Cc1n[nH]c(=NC(=O)c2csc(NC(c3[nH]nnc3C)=O)n2)o1 CN1C(C(N2CCN(C3CCN(C(=O)C=CC4CC4)C3)CC2)=O)CCS1(=O)=O Cc1ccc(CC(=O)NNC(=O)NC2CN(C)CC2O)c(C)c1Br C1(C(N(CC(C)NC(c2cc(C)n(CCO)n2)=O)CC)=O)CC2CCC1C21CC1 n1(CC(=O)N(CCC)Cc2c(Cl)oc3ccccc23)cnc2ccccc2c1=O N1(C(C(CC(C)C)NC(=O)C(C#N)C(C)C)=O)CCCC2CN(C)CC12 C(C)(C1=CCN(C)CC1)NC(CCN(C(c1c(C)nncc1)=O)CCO)=O N(C(=NCCC(=O)NC1(C(=O)NC)COC1)NCC(C)(C)C(=O)OC)SCC N1(C(CCC)=O)CCCN(C(c2cccs2)=O)C(C(C)C)C1.c12cccc(c1)C(=O)CS2.N CC(C)CC(C(=O)NC1CN(C(c2csc(Cl)n2)=O)CC12CC2)C(C)C c1(OC)cc(C(=O)NC2CCN(C(C3C=CCC3)=O)C2C)sc1Br c1(OC)ccc(C(N2CCCC(F)(C)C2)=O)cc1CNC(=O)C(CO)N(C)C.C(N)=O.N N1(N(CC(C)C)C(=O)C=CC(C)(C)NC(c2ccsn2)=O)CCC(C(N)=O)C1 C(c1cccs1)=CC(=O)NC1C(C(N2CC(C(=O)NCCO)C2)=O)C1(C)C Cc1[nH]c(=N)sc1C(=O)NC1(CNC(C2C3CC3C3CC23)=O)CC1 CC1(C)C(=O)CC1C(=O)NCCC1CN(C(=O)CC2(C)CC2(F)Cl)C1 CC(C)C1=CCC(C)(NC(C2CC(c3cccc(Br)c3)C2)=O)CC1 Cc1scc(C(=O)NC2CCN(C(=O)C(C)NC(C3CCCC3)=O)C2)c1C C1(NC(CCN(CC)CC)=O)CCC(NC(C2(COCCC)CC=CC2)=O)CC1 C=C(C)C(CC(=O)NCC(C)(C)OC1CN2CC1CNC2=O)OCC.SCC c1(C(N2CC(CC)C(NC(=O)CC3C(=O)NN=C3C)C2)=O)ccc2ccoc2c1 c1(C(=O)OCCn2cc(-c3c(Cl)ccc(OC)c3)nn2)nc2c(C)cccc2[nH]1 CON=Cc1ccc(C(=O)Nc2cc(Cl)cc(F)c2F)cc1 N1(C(C2=NNC(=O)C2)=O)CC2CN(C(c3cccc(CO)c3)=O)CCC2(CO)C1 c1(C(N2CCCC(CCNC(CC(=O)NCC#C)=O)C2)=O)ccc(NC)c(F)c1 C(=O)(CC(O)C(Cl)(Cl)Cl)N1CC(O)(CNC(c2sccc2C2CC2)=O)C1 CCCCC(C)CCC(=O)N1CCCC(C)(C)C1C(=O)NCC12CCC(CC1)C2 CON(CCC(=O)N1CCCCC(C)(C)C1)C(=O)C1(C)CC2CCC1O2 CC(CCC(=O)NCCCNC(=O)C=CC(C1CCCC1)=O)c1ccccc1 c1(C(C)NC(c2ccc(C(N)=O)[nH]2)=O)nocc1C(=O)NC1CC1F C1(C2CCOCC2)(C(N2C(CN3C(=O)CCCC3)CCC2)=O)CC1 c1(OCC)cc(Cl)cnc1C.C1(=O)C(C)N1.C1C(C)N1CC(=O)NC(N)=O C1(NC(c2cncc(F)c2)=O)CCN(C(c2c[nH]nc2C(F)F)=O)CC1F C1(NC(CC(CCSC)O)=O)CN(C(c2cccc[n+]2[O-])=O)CC12CCOCC2 C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(c2cc(C3CCC3)on2)=O)CCC1 C1(C(N(C(CC)C)C)=O)(COC)C=CCN1C(c1cncc(C)c1)=O c1(C(=O)NC2CC(NC(c3c(C)n[nH]c3)=O)C2)cc2c(Cl)cncc2s1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)N1C2CN(C(C3CCC(C)C3)=O)CC21 C(C1c2ccsc2CCN1C(c1nocc1Cl)=O)NC(c1ccc(OC)cc1)=O O=C1CC(CC(=O)NC23CC(CNC(C4C(F)(F)C45CC5)=O)(C2)C3)=NN1 CC(C)CS(=O)(=O)CCC(=O)NCC(C)(C1CC1)NC(=O)CC(=O)OC(C)(C)C C(=O)(C1Cc2ccc(F)cc21)N(C)CC1CCCN1C(c1cc(C(N)=O)c[nH]1)=O C=CCC(CNC(C1CC1C(C)(F)F)=O)NC(=O)C(C)=C(C)C C(CCC(C)C(=O)NC1CN(C(c2ccc(Br)nc2O)=O)CC1O)OC c1(C(=O)NC(CC(C)C)CNC(=O)CC2CC(=O)C2)cc2c(nc1O)CCCC2 C1(CNC(CCC=CC(C)C)=O)(CO)CCCN(C(C2CCCC23CCC3)=O)C1 CC1(C)CCCC(O)(C(=O)NCC2CC2NC(=O)CCn2cncn2)C1 Cc1cc(C(=O)NCc2cn(C3CN(C(=O)COC4CC=CC4)C3)nn2)n[nH]1 N1(CC(=O)NCCC(C)N(C)C(c2ccc(F)cc2F)=O)CCn2ccnc2C1 C=CCC(C(=O)NCC(C)CC(=O)N1CC(F)CC1C)OC C(CCCCC(C)(C)N)NC(c1ccc(C)nc1)C(=O)OC C(CC(C)C(=O)NCC1(F)CC(NC(c2cccc(C(C)(F)F)c2)=O)C1)OC C(Cc1ccco1)(C(=O)NCC1CCC1C)NC(CN(C(C)=O)C)=O Cc1c[nH]c2ncc(C(=O)NCC3(C)CCCN3C(=O)CCC(C)C)cc12 c1(OC)cc(C)c(C(=O)NCC(C2CCOC2)NC(c2cnc(S)[nH]2)=O)c(C)c1 c1(C(=O)NCC2CN(C(c3[nH]n(C)c(=O)n3)=O)C(C)(C)C2)ccc2c[nH]nc2n1 N1(c2ccnc(C)n2)CCC2(NC(=O)CC(C3CCC3)C3CCC3)CCCC12 CC(CC(=O)N1CCC(OCCNC(C2CC(N(C)C)C2)=O)C1)C(F)(F)F Cc1noc(CNC(c2ccn(-c3ccccc3)n2)c2nnnn2C)n1 C(=O)(C(O)CC(F)(F)F)NCC1CC(F)(CNC(C(C)NC(CC)=O)=O)C1 Cc1c(C(=O)NCC2C(C)CCCN2C(=O)C=C2CCSCC2)sc2cncn12 C1(C(N2C(C)CC(NC(c3ncncc3Cl)=O)C2)=O)(CF)CC2(CCC2)C1 CC1C(=O)NNC(=O)N1.C1(C(N)=O)CC2CC(C1)C2 C1(CNC(C2C(CC)CCO2)=O)CC(F)(F)CN1C(=O)CCC(=O)N(C)C C1(NC(C2CCCN2C(=O)CCOCCCOC2CC2)=O)CC2CCC(C1)S2(=O)=O Cc1ccccc1-n1ccc(CN(C2CC(c3ccccc3)C2)C=O)n1 CCCC(C(=O)OC)C(=O)NCC1(CNC(C2CCCCC2O)=O)CCCC1 Cc1cc(C)c(C=CC(=O)NCCC2(NC(=O)CC3CCCC3C)CC2)c(C)c1 N1(C(CN(C2CCCC2O)C)=O)CC=C(CNC(C2(F)CCOCC2)=O)CC1 N1(CC)CCOCC1(C)c1cn(CCCCF)nn1.C12(CCC1)CCNC2=O c1(-n2cc(C3(NC(=O)CO)CC(F)C3)nn2)ccccc1F C12(N3C(=O)COC3=O)CC(OC)C1C2.c1(O)ccccc1.CC C(=O)(C1CCc2cccc(O)c21)NCC1N(C(C23OC(C)(C)C(CC2)CC3)=O)CC1 CC1C(NC(=O)C(C)(C)C(F)F)CC2CCC1N2C(=O)CCN1CCCC1=O C(=O)(CC(C)CN=c1[nH]c(N2CCC(C(F)(F)F)CC2)nc(=N)[nH]1)NC C(=O)(CC(C)C(C)(C)C)N1CC(C)(NC(c2ccc(C(C)C)o2)=O)C1 Cc1ccc(C(=O)NCc2nc(CNC(=O)CCC3CC3C)cc(O)n2)c(Cl)c1 CC(C)C(O)CC(=O)N1CCN(C(=O)Cc2cncc(F)c2)CC1CCO C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CCOC)(NC(c2c(CC)non2)=O)C1 C12(CNC(C3(F)CN(C(c4cc(C)n(C)n4)=O)C3)=O)CCC(C1)C(=O)N2 C(=O)(n1ccnc1C(=O)NC1CCCC1NC(C12CC(O)C1C2)=O)OC(C)(C)C C1(CCC(=O)N(C(C)CNC(c2oncc2C)=O)CC)CCCN1C CC(C)CC(CO)N(C(=O)C(c1ccccc1)NC(=O)C(C)N=[N+]=[N-])C N1(C(c2ccc(C(C)=O)o2)=O)CCN(C(=O)C(C)(C)CC(F)F)CC(O)C1 C1(NC(c2sccc2C(F)F)=O)CCN(C(C2CC3CCC2C3)=O)CC1CO N12CCCC(C1=O)C2=O.N1(C(c2ccccc2)=O)CC2CCCC12.C(=O)(CCO)OC CC(C)CCC(=O)Nc1ccccc1C1CCN(C(=O)OC(C)(C)C)CC1 c1(OC)ccc(S(=O)(=O)Oc2cc(Br)c(C#N)cc2Cl)c(C)n1 C=Cn1nncc1C(N1CCCCC1CC(=O)NC(CC)CCOC)=O CN1C(=O)CCC1CC(=O)NCC1CCCN1C(c1cc(C(F)F)n(C)n1)=O C1(CCC(N2CCC(C(C)NC(Cc3ncc(CC)[nH]3)=O)C2)=O)CCC(O)CC1 CC(C)C(C#N)C(=O)N(C1CN(C(c2nn(C)cc2Cl)=O)CC1(C)C)C c1(OC)ccc(C(=O)NC2CCC2NC(=O)Cn2cnnc2O)c2c1CCCC2 c1(C(=O)NCCOCCNC(C(c2ccccc2)C)=O)cc2c[nH]nc2s1 C1(NC(CC=CCC)=O)CCN(C(=O)C(C)=C2CC2)CC1C C1(C2CC2)(NC(=O)CCc2ccccn2)CCN(C(C2CCC(=O)N2)=O)C1 C1(C(=O)NC2(CNC(=O)CCc3ccon3)CCCC2)CC2(CCOC2)C1 N1(C(c2cc(OCC)n[nH]2)=O)CCCC(NC(C2CCC=CO2)=O)CC1 C(=O)(C(F)CCC(C)C)N1CCCCC(NC(C(CCC)CN(C)C)=O)C1 CC(C)C(C)CCNC(C1OCCC1CNC(=O)C=Cc1cc[nH]c1)=O C(=O)(CC(C)(C)CC(F)(F)F)N1CC=CC(NC(C2(COC(C)C)CC2)=O)C1 Cc1cc(C(=O)NCC2CC(NC(c3[nH]nc(C(F)F)c3C)=O)C2)cn(C)c1=O c1(C(=O)NCC(CC)NC(=O)CC2CCC(C)(CC)O2)c(F)ccc(C#N)c1F N1(C(c2c(C(C)C)n[nH]c2)=O)CC2(C(=O)NCCC3(O)CCOC3)CC1CO2 Cc1cnn(C)c1C(=O)NC(C1CCCCC1)CNC(c1ccc(Cl)cc1)=O N1(CC(O)CC2CCOCC2)CC2CC3CC2C1C3C(F)(F)F c1(Cc2nnc(CNC(C(N3C(CC(C)O)CCC3)=O)=O)s2)cccc(F)c1 c1(C(N2CCCC(CNC(CCNC(N)=O)=O)C2)=O)ccc(F)c(C(F)F)c1 C1(CC(=O)NC(CCC)c2ccco2)CCN(C(=O)C(C)SC(C)C)C1 Cc1ccc(N(C2CCN(C(C3CCOC(C)C3)=O)C2)C)nn1 C1(O)(C(N2CC3C(CNC(c4ncc(OC)cn4)=O)(C3)C2)=O)CN2CCC1CC2 N1(C(COC(CC)C)=O)CC(NC(=O)CC2(n3ccnn3)CC2)C(C)(C)C1 C(CC(CNC(C1(OC)CCC1)=O)NC(c1cc(-c2ccccc2)co1)=O)OC C1(NC(NCc2nnc(C)s2)=NCCN2CCCC2)CN(C(C)=O)CC12CCC2 C(C)(C(C)C(=O)NCCCC1(O)CC1)NC(CC(=O)NCC#C)=O c1(CNC(=O)CCc2ccsc2)ncccc1NCc1ccc(C(=O)O)[nH]1 C1(C)(C(=O)NC(CCOC)C)CC(NC(=O)CSCCOC)C1 Cc1c(NC(C)C(C2CCCCC2)NC(=O)Cc2nccs2)ncnc1C(C)C C12(CNC(c3n[nH]c(C)c3F)=O)CCC1CN(C(c1ccnn1C(C)(C)C)=O)C2 n1(CC(=O)NCCCOCCOCCNC(C2C(=C)C2)=O)ccc(C)cc1=O N1(C(c2cc(C)c(C)[nH]2)=O)CCN(C(=O)CN2CCN(C(N)=O)CC2)C2CC12 C12(C(N(CCCO)CCC)=O)CCN(C(c3nonc3C)=O)CCC1C2 C1(NC(Cc2c(C(C)C)cccc2)=O)CC2CC1CN2C(=O)CC(C)(C)C C1(NC(c2ccc(OC)nc2C)=O)CCC2(CCN(C(=O)CCNC(N)=O)CC2)C1 C(=O)(C1CCCn2nccc21)N(CC(CNC(Cc1c(C)noc1)=O)O)C CCC(CC(=O)NCC1CC(CF)C1)NC(=O)C(CC)N(CC)CC Cn1c(O)nc2cccc(C(N3CCC(NC(=O)CC4CCOC4)C3)=O)c12 N1(C(C=C(COC)C)=O)CC2CC(NC(c3ncc(C)cc3Br)=O)C1C2 N1(C(CCC(=O)NC)=O)CCC(C2(O)CC(NC(C3CC3C(N)=O)=O)C2)CC1 C1(SCC)CN(C(=O)CN(C)C(C)=O)CCN1C(c1ccnc(C2CC2)c1)=O C1(C)(NC(C(CC)OCC)=O)CCCCC1C(=O)Nc1cncc(C2CC2)c1 N1(C(C2OCC(C)C2)=O)CCN(C)C(C(N2CCC(CCO)C2)=O)C1 N1(C(C(Cc2cn[nH]c2)NC(CNC(=O)NC)=O)=O)CC2CCC1C(O)C2O CC1(C)NC(=O)CC1C(=O)NC1CCC(NC(c2cccc(C3CC3)c2)=O)CC1 N1(C(C2N(C(C)=O)CCOC2)=O)CC2CCC1CN2C(=O)CC(C)(C)C1CC1 C1(NC(c2cccc(C(=O)NC)n2)=O)CN(C(=O)C(F)OC)CC1(C)C C1(C(N2CCC(C(=O)NC3(CC)CN(C(N)=O)C3)CC2)=O)CC2CCCC2C1 Cc1cc(Cl)c(Cl)cc1C(=O)N(C)C.N12CCN(C(=O)OC(C)(C)C)CC1C2=O N1(C(c2cccc(OCCC)c2)=O)CCC(CNC(=O)CC(C)OC)C12CC2 c1(CCC)ncc(NC(C2CC(NC(=O)CN3CC(=O)NC3=O)C2(C)C)=O)cn1 c1(C(=O)NC(C)(CNC(C2CC2(C)C)=O)Cn2cccn2)cc2c[nH]nc2s1 C1(SCCNC(C(C=C)O)=O)CCCN(c2ccncn2)C1 c1(C(N2CC(OC)C(O)C2)=O)cnc(O)c([N+](=O)[O-])c1.n12cnc(n1)CC2 CC1CC(C(=O)NCC(C2CC2)N(C)C(c2cncn2C2CC2)=O)CO1 CC1CC(C(=O)NCC23CCC(CC2)N3C(c2ccoc2Cl)=O)CCC1=O Fc1cccc2c1OCC(Nc1nccc(=NCSCCC3CCC4CC34)[nH]1)C2 C(CCCCCC(=O)O)NC(=O)OC(CCN(CC=C)CC=C)=O Cc1c(C(=O)NCCC(C)N(C)C(C2(F)CCOC2C)=O)cnn1C C1(C(=O)NC(CCC)CO)(OC)CCN(C(c2cc(C3CC3)on2)=O)C1 C(=O)(C(F)C(C)CNC(=O)Cc1cc[nH]n1)N(C(C)C)CCO C1(CC(=O)NCC2(OC)CN(C(c3[nH]cnc3C)=O)C2)CC(=O)NC1=O C1(=CC(N2CCCC2CNC(=O)C=CC2CC2)=O)CCSCC1 N1(c2ccnc(COC)n2)CCCC12CCN(C(=O)C(CCSC)OC)C2 CCCC(C(O)C(=O)NCC1(CC(C)C)CCC1)NC(=O)CCC1CCOC1 CC(C)(C)CC(=O)N1CCC(C(C)(C)NC(C2(CO)CCCCO2)=O)C1 C1(NC(CSCC=C)=O)CC12CCN(C(=O)C(c1cccc(Br)c1)C)CC2 CCCCCC(CC)C(=O)N1CC(CC(=O)NCC(C)(C)C(F)(F)F)C2(CC2)C1 C#CC1(C(=O)NC2(COC)CCC2)CN(C(=O)C(CCC)N(C)C)C1 C(CS(=O)(=O)NCc1cc(C(C)(C)C)no1)(C1CCOCC1)OCC C(C(C)C(=O)N(OC)C(C)C)N1CCN(C(C(CCCC)=O)=O)CC1 c1(C(N2CC(O)CC(NC(CC(C=C)(C)C)=O)C2)=O)ccc2ncncc2c1 CC1CC(CCNC(C2CS(=O)(=O)C2)=O)CCN1C(=O)Cn1nnnc1C1CC1 N1(C(c2cn(CC=C)nc2)=O)CCC(CN(C(=O)C(C)(O)COC)C)CC1 c1(NCCCc2cccc(OC)c2)nc2c(cc1Br)CCC2O c1(C(=O)NCC2OCCN(C(CC3(C)CC3)=O)C2)nccc2n[nH]cc12 C(C(CC(=O)N1CC[Si](C)(C)C1)NC(c1cnsn1)=O)OC C1(CC(=O)N(CCNC(CCCCN(C)CCO)=O)C)Cc2ccccc2O1 Cc1cc(C(=O)NCC2CCN(C(=O)C(C)n3cncn3)C2)c(N)c(F)c1 c1(C(N2CC(CNC(=O)CCC3CCCC3)OCC2)=O)ccc2c(c1)COB2O c1(C(=O)NC2CC3CC2N(C(=O)C=Cc2ccco2)C3)ccc(Cl)c(F)c1F C(C)(C)(CCCCC(=O)N1CC(O)CC1CNC(c1ccn(C2CC2)n1)=O)OC C#CC1(C)CCN(C(=O)CCCCCNC(=O)CSC(C)(C)C)CC1 c1(C(N2C(CNC(C(COC)OC)=O)CC3CC32)=O)cnc(OC)c(C)c1 c1(C(N2CC(NC(CSCCC)=O)C(O)C2)=O)c(O)nnc2c1CCC2 c1(CCC(=O)NCCC2CC(NC(C=CS(C)=O)=O)C2)nnc(S)nc1O C1(NC(C=CC=CC)=O)CC2CC(NC(=O)COc3ccc(C)c(C)c3)C2C1 C=CC(C)(O)CC(=O)NCC1C(C(=O)Nc2nn(Cc3ccccc3)cc2C)C1 N1(C(C2N(C(C)=O)CCC2)=O)C2CCC1CC(N(C)C(C1(C)CCCCO1)=O)C2 CC1CN(C(C2CCCC3CC23)=O)CCN1C(c1ccnc(F)c1)=O N1(C(c2cc(C(N)=O)[nH]n2)=O)CCCC(NC(C2CCS(=O)(=O)N2)=O)C1 C(=O)(CC(C)(C)N(C(C12CCC(CC1)C2)=O)C1CC1)N(C)CC1C(C)C1 c1(C(c2n(C(C)C)nnn2)NCc2nc(C(C)(F)F)cs2)ccccc1C1CC1 C1(NC(C(COC(C)C)NC(=O)OC(C)(C)C)=O)CCC(=O)NC1=O C1(C(=O)NCC(CO)NC(c2c(NC(C)=O)cccc2)=O)CN2CCCN1CC2 c1(CSCC)cccc(C(=O)NC2CN(C(=O)CCc3nc(O)n[nH]3)C2)c1 C1(C(=O)Nc2cc(Br)cnc2Br)CC2(CC2)CN1C(c1cc(Cl)c(Br)s1)=O N1(C(C(C(CC)O)C)=O)CCC2(C1)CN(C(=O)CNC(=O)C(F)(F)F)CCO2 N1(C(C2(CC)CCCN(C(C3CCCSC3C)=O)C2)=O)CCCC(C)(C#N)C1 C(C(=O)NCC(CO)C(C)(C)C)(C(C)(C)O)NC(c1c[nH]c(=NC)s1)=O C1(CC(=O)NCCN(C(=O)CCc2cnc(O)[nH]2)CC(C)O)CC2C=CC1CC2 C(=O)(C(F)(F)CN(C)C)NCC1C(Cn2cc(CC(C)C)nn2)C1(F)F C1(N(C(COCC)=O)C)CN(C(c2cc(C#N)cn2C)=O)CC12CC2 C1(NC(CC=C)=O)CN(C(=O)CC2CC3CCC2CC3)C2CCCCC12 c1(C(=O)NCC2(C(N3CCC3N3CCCCC3)=O)CC3(CC3)C2)ncc(F)cn1 CCCCC(C(=O)N1CCCOC(C(C)C)C1)NC(=O)Cc1ccn(CC)n1 N1(C(C2CC(C)(C)OCC2)=O)CCC2CC1CN(C(c1ccon1)=O)C2 CCC(C(=O)NCC(C)(C)NC(=O)C(C)(C)OCCOC(C)=O)OC C1(C(=O)NCc2cc(C(N(C3CCC3)CC)=O)sc2)CC2(C1)CC21CC1 c1(C(N2CC(F)CC(C(N3CC(C)C(O)CC3)=O)C2)=O)cccc2c(O)nccc12 N1(C(C2C(C#C)C2)=O)CCCC2(C1)CN(C(c1scc(C)c1Cl)=O)CCO2 N1(C(C(CCCNC(=O)CC2CC2C2CC2)O)=O)CCCC12CCOC2=O C1(C)(CNC(C(C)NC(=O)C2CC2)=O)CCCN(C(c2cnc(C(F)(F)F)s2)=O)C1 N1(C(c2cc(C)c(O)cc2)=O)CC(CNC(=O)CC2(O)CCC2)CC12CCC2 CCC(O)C(C)C(=O)NC12CC(NC(c3cnc(-c4ccco4)s3)=O)(C1)C2 C1(CC)(NC(C2C3CCCOC23)=O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1 N1(C(C(CO)OC)=O)CCC2CN(C(=O)C(C)(C)OC)CC12 O(NC(=O)C(CCF)NC(C1CCC(C)(C)C1)=O)CCOCC#C c1(C(=O)NCC(CC)NC(C2(C#N)CC=CC2)=O)c(OC)ccc2ncccc12 c1(C(N2CC(C(=O)NCc3n[nH]c(C)c3Cl)(CC)C2)=O)ccc(C)nc1O C#Cc1ccc(CC(N2CCC(C(F)C(=O)NCC(C)(CO)CO)C2)=O)cc1 N1(C(C2(OCC)CCC2)=O)CCC2CC2(C(=O)NC2(C)CC3(CCC3)C2)CC1 c1(C(N2CC(CN(C(C(n3ccc(C(F)(F)F)n3)C)=O)C)C2)=O)ccnc(O)c1 Cc1nc(=N)[nH]c(C)c1C(N1CCC(CCNC(=O)Cc2ccc(F)cc2)C1)=O CC(C)(CCC(=O)NCCN1CCCC(O)C1)NC(c1nc[nH]n1)=O c1c(O)cc(NC)cc1O.N1(C(C)=O)CCN(c2cc(N3CCCC3)ncn2)CC1 C1(CN2C(CC(c3ccco3)=O)CCCCC2)CCCC2(CCC2)O1 C1(CN(C(=O)Cc2cc(=O)n(CC(C)C)[nH]2)CC)CC12CCN(CC(O)CO)CC2 c1(C(N2CCN(C(CCSC)=O)C(C3CC3)C2)=O)cc(Cl)c(OC(F)F)cc1C C1(n2cc(-c3c(C(=O)OC)n[nH]c3)nn2)CCCN(Cc2cncc(C)n2)C1 CC1C(NC(=O)C(O)Cc2ccccc2Cl)CCCN1C(c1cncc(Cl)c1)=O c1(CC(C)NC(C(=O)N(C)Cc2cn(CC(C)C)nc2)=O)csc2ccccc12 c1(OC)cccc(Cc2nc(-c3cncnc3)nn2-c2cncc(C)c2)c1Cl N1(C(Cc2cc(C)on2)=O)CC(CNC(c2cccc(O)c2F)=O)CC12CCC2 C1(CC(=O)NCCCN(C)C(c2cnc(C(F)(F)F)n2C)=O)SC(=N)NC1=O c1(NCCc2cnc(CC)s2)ncccc1S(=O)(=O)NC1CC1c1ccco1 c1(OC)ccc(OC)c2sc(=NCC(O)CNC(c3n[nH]c(O)n3)=O)[nH]c12 c1(C(C(=O)NCCNC(c2ccc(F)cc2)=O)O)cccc(F)c1 C1(C(=O)NCC(O)CN(C)C(c2cc(Br)no2)=O)(OCC)CCOCC1 C1(NC(c2cccc(SC)n2)=O)CC2CCC1CN2C(=O)C(CC(C)C)N(C)C c1(CCNC(=O)NCCN2CCCC(CC)C2)cc(O)nc(O)n1 C1(N(C(c2c(OCC)ccs2)=O)CC)CCCN(C(C2(C#N)CCCO2)=O)CC1 C=CCCC(F)(F)C(=O)N1CCCC(CC(=O)NCC=CCCC)C1 c1(NC(=O)NC(CCC)C)nccc2cncn12 N1(C(c2occ(C)c2)=O)C(C(=O)NC2(c3ncccn3)CC2)CCC1C1CC1 N1(C(C2(C(=O)OC)CC2C)=O)CCC(n2cccn2)(CNC(=O)C(C)C)CC1 NS(=O)(=O)c1ccc(C(=O)NC2CCC(NC(c3ccc(F)c(O)c3)=O)CC2)s1 N1(C(=O)Nc2cn(CC)nc2C)CCC2CCCCC12 C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCC(N(C)C(C2CCCN2C)=O)C1 c1(C(C(=O)NC(CC2CN(C(C(C3CCC3)OC)=O)C2)C)C)c(C)nn(C)c1C C1(C)(C(=O)NCC(CN(C(C(C)O)=O)C)C)CC2CCC1CC21OCCO1 c1(C2(C(N(C(CNC(CNC(COCCOC)=O)=O)C)C)=O)CC2)cccnc1 CCCCC(C(=O)N1CCC(C2CC2NC(=O)C2=COCCC2)CC1)C(C)C c1(OC(C)C(N2CCC(O)(c3cccc(C(=O)O)c3)CC2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2CC(NC(C3(C#N)CCC3)=O)C2)cncc2nc[nH]c12 c1(CC(=O)NC2CCN(C(C(F)=C(C)C)=O)CC2(C)C)cc(S(N)(=O)=O)cn1C CC(c1ccccc1Cl)=CC(=O)NCC1CCC2(CN(C(=O)CC)C2)O1 C1(CC)CN(C(=O)CCCC(F)F)CCN1C(c1ccc(Cl)c(F)c1)=O C(CNC(c1cccn1CC)=O)(C(C)C(C)C)NC(c1c(CC)onc1)=O C(=O)(CC(C)C(F)F)NCCOCCNC(C(C)Oc1cccc(CO)c1)=O N1(C(C=Cc2nc(C)sc2C)=O)CC2CCN(C(C3CC(C)(O)C3)=O)CC12 N1(C(c2cc(C)no2)=O)CC2CCC2(C(=O)Nc2ccc(Cl)cc2)C1 N1(C(Cn2c(=N)nc[nH]2)=O)CCC2CN(C(=O)Cc3ccnc(Br)c3)CCC12 CCC(CC1CC1)CC(=O)NCc1ccsc1C(=O)NC(c1ccccc1O)C C1(CN(C(c2cc(C(N)=O)cn2C)=O)CC)CCCN(C(=O)C=CC2CCC2)C1 CC1CCCCC1(CNC(c1sccc1F)=O)NC(C1(n2ccnn2)CC1)=O N1(C(CC(OCC)OCC)=O)CCCC2(C1)CN(C(c1occc1Cl)=O)C2 C1(C(=O)NCCN(C(=O)C(F)n2cccn2)CC)CCCC12CCC2 N12CCN(CC1)C(=O)NCCOC(=O)C2C.C(C)(C)(C)OCC c1(C(N2CCN(C(CC=C)=O)CC2CC#N)=O)cccc([N+](=O)[O-])c1O C1(NC(c2ccc(C)cc2)=O)CN(C(C2(C#N)CC2)=O)CC2(CC2)C1 c1(CC)nccnc1C(=O)NN(C1CCCN1)CCC1CCCCC1 Cc1c(C(=O)NCC(CNC(C2(F)CCC2)=O)C(F)(F)F)oc2ccc(F)cc12 N1(C(C(C)OC)=O)CC2CCC2(NC(=O)Cc2ncc(C)s2)C1 C(N=c1ccn(C)[nH]1)(c1ccn(C)n1)C1C(CN(C)C)C1 Cc1cc(N2CC3C(CNC(C45CC4C5)=O)C3C2)nc(S(C)(=O)=O)n1 c1(NC(CCNC(C(C)OC(F)F)=O)=O)ccc2c(c1)NC(=O)C2 C(=O)(C(CC)CC(C)C)N(C(C)C(N1CCC(O)CC1CC)=O)CCC c1(OC)ccc(CCC(=O)NCC(CNC(c2ccc(SC)[nH]2)=O)OC)cc1 Cc1nn(C)c(C)c1CC(N1CCC(C)C(NC(=O)C=Cc2cn(C)cn2)C1)=O N1(C(c2cc(Br)c(F)cc2O)C(=O)NC(CC)C)CCc2cccnc2C1 c1(C(N(C2CCN(C(=O)COC(F)(F)F)C2)C)=O)ccc(C(F)F)nc1 Cc1cc(C(=O)NCC(C)NC(=O)C(C)(C)c2cnn(C)c2)nc(O)c1 c1(-n2c(C)cc(C)n2)ccc(NC(=O)C(=O)NC2CC(=O)N(C)C2)c(F)c1 CC(CCC(=O)N1CCC2CC12C(=O)NCCOCCC1CC1)N(C)C C1(C)(C(N2CCC(CNC(C(C)(Cl)Cl)=O)C2)=O)COC(=O)O1 CCC(CCC(=O)NC1(C(=O)NCCC2CCCC2)CCSC1)OC CCC(C)CCCC(=O)N1CCC(C(=O)NC(C)CSC(F)F)CC1(C)C C1(C(N2CC(N(C(=O)CC3(N(C)C)COC3)C)C2)=O)(OC)CCSC1 CN1CCC(NC(c2n[nH]c3c2CN(C(C2CC=CC2)=O)C3)=O)C(C)(C)C1 c1(CC(=O)NC2C(F)CCN(C(C(CCC)C)=O)C2)c(C)cc(OC)cc1C C1(C(=O)OC)COCC1c1ccccc1.C1(C)C(=O)N1CCF.C1CNC(=O)N1 CC1CCC(O)(C(N2CCC2(CC(C)C)CNC(c2cnc(N)cn2)=O)=O)CC1 C(=O)(CCCC(=O)N(C)C)N1CCC(C)(C(=O)NCC2(OCC)CCOC2)C1 Cn1c(Cl)cnc1CNc1cc(NCC2(C)CS(=O)(=O)C2)ncn1 c1(CCC)ccc(N)c(C(N2CCN(C(=O)C(CO)NC(N)=O)CC2C)=O)c1 N1(C(=O)NCc2c(OC)cc(Br)cc2)CC(CO)C2(CCOCC2)C1 Cn1cc(C(N2CC(O)(CNC(C3CCC3C(F)(F)F)=O)C2)=O)nn1 c1(C(N2C3CCC(NC(=O)C(Cl)=CCl)C(C3)C2)=O)cccc2nc(O)ccc12 c1(OC)cnc(NC(=O)CC2C(C)CCN2C(=O)OCC2(CO)CCCC2)cn1 C1(CNC(c2ccc(CC)cc2)=O)CC2(CCC2)CN1C(C1CC1F)=O C1(OCC)CC(CNC(=O)C(=O)Nc2ccnc(C(C)C)c2)N(C)C1 c1(C(=O)NC2CCN(C(C3C(C)CCC3)=O)CC2)cc(C(F)F)cc(Cl)c1 N1(C(C2C(C)(COC)C2)=O)C2CCCC1CN(C(c1ccc(Cl)c(Cl)c1O)=O)C2 C(C(C)(C)C#CC(=O)NCc1cccnc1F)NC(CC(C)F)=O c1(C(=O)NC2(CN(C(c3scc(OC)c3)=O)C)CC2)ccc(C)nc1 O=C(CC=C(Cl)Cl)NC(c1cccnc1)C(=O)NCCOC(F)F C#CCCCCCCC(=O)NCC1COCCN1C(=O)C(C)CS(C)(=O)=O Cc1cccn2cc(C(=O)NC3CC(F)CN(C(c4c[nH]c(=O)cn4)=O)C3)cc12 C(=O)(C(CC(C)C)ONC(=O)C(C)NC(N)=O)NCc1cnc(C)[nH]1 Cc1cc(C)c(C(N2CC(O)CC2C(=O)NCc2cc[nH]n2)=O)c(C)c1 C1(O)(CNC(C2CC(C)C2)=O)CCN(C(c2csc(-c3ccoc3)n2)=O)C1 N1(C(=O)COC2CCCC2)CCCC12CCC(NC(C13CSC(C1)C3)=O)CC2 c1(C(=O)NC2CC(C)N(C(=O)CN3CCS(=O)CC3)CC2)ncsc1S(N)(=O)=O C=CCC(CNC(=O)C=C(C)C(C)(C)C)C(=O)N(CC(C)C#N)C1CC1 C12(C(CNC(c3nc(N(C)C)co3)=O)NC(c3c(C)snn3)=O)CCC(CC1)C2 C1(C(=O)OC)CCCCC1(C)NC(=O)CCCn1cc(CC(C)(C)O)nn1 c1(C(=O)NC(CCOC)CO)coc2c1CN(C(=O)CCc1cnco1)C2 C1(CCC(=O)NCCCN2CCC2)CCCN(C(c2cnsc2)=O)C1 N1(C(C)=O)CC2CCC1CN2C(=O)C(F)F.c12ccc(o1)C(=O)NC2 c1(CN2CCC(CCC#C)C2)nc(C2CC2)n2ccccc12 C1(O)(C(=O)NCc2cc(C(=O)NCC=CCOC)no2)CCCCC1 N1(C(C(C)(C2CC2)OC)=O)CC(CNC(c2cn(C3CCOC3)nn2)=O)C(O)C1 c1(C(=O)NCC(CC(C)C)(C)NC(C2CCN(C)CC2)=O)ncc2ccccn12 c1(N2C(C(C)(C)NC(C(C)OCCOC)=O)CCC2)c(C)cccc1[N+](=O)[O-] N(C(=NCCc1ccoc1)N1CCS(=O)(=O)C(C)(C)C1)C(CC)C c1(OCC=C)ccc(C(=O)NCC2(NC(=O)C(C)CC(C)C)CCC2)cc1OC N1(C(C2C(CCC)CCC2)=O)CCC2CCN(C(c3ccc(F)cc3C)=O)C2C1 c1(C(=O)NCC(CC)NC(=O)CCc2cncs2)cnc(O)c2ccsc12 C(=O)(CC=C(Cl)Cl)NCC(N1CCN(C(C2CCCOCC2)=O)CC1)(C)C c1(C(=O)NC(C2CN(C(C3(C)CC3C(F)(F)F)=O)C2)C)cc(C#N)c(F)cc1F C1(C(=O)NCC(c2cccnc2)NC(=O)CO)C2CCC1(c1ccc(F)cc1)C2 Cc1ccnc(C(=O)NC2(C3CCCN3C(=O)CCCc3n[nH]c(=N)s3)CC2)c1 CC(C)CC(C)(O)C(=O)NCc1ccc(C(=O)NC2CC(C)CC(C)(C)C2)nc1 N1(C(CC=CC=C)=O)CCN(C(c2cnc[nH]2)=O)C(CCCC)C1 c1(-n2cc(C3(C)N(C(C(CCC)F)=O)CCC3)nn2)ccc(C#N)nc1 Cc1ncc(F)c(NC2CC3CN(C(C4(C)CNC(=O)C4)=O)CC23)n1 n1(CC(=O)NCC2C(NC(=O)CCC3CC3)CCCC2)cccc([N+](=O)[O-])c1=O N1(C(C(CC(C)=O)C)=O)CC(C(=O)NCc2ncnn2C)C2(CCC2)C1 N1(C(c2c(OC)cccc2)=O)C2CC1CN(C(=O)Cc1ccc(C)o1)C2 n1(CC)cc(C(C)NC(=O)C(C2CN(C(C3C=C(C)CS3)=O)C2)OCC)cn1 C(CN=C(NC1CC1)NC1CC(=O)N(C2CC2)C1)(C1CCCCCC1)OC c1(NC(C=CCN(C(C=C(CCC)C)=O)C)=O)ccc(F)cc1CO C(=O)(CN=c1c(C)c[nH]cc1C)N1CCCC(CNC(C(CC)C(C)C)=O)CC1 c1(OCC)ncccc1NC(C1CCN1C(=O)NCCC(=O)NC(C)(C)C)=O N1(C(C(CC#CC)NC(C2CCCCNC2=O)=O)=O)CCOC(C)(C)C1C C(=O)(C(C)CC(=O)NCC(C)C(F)C(=O)Nc1cc(C)ccc1OC)OC C1(C(=O)NCCC(F)F)CCCSC1C.C1C(=O)N(C(C)C)CCN1C C(=O)(C(CC(C)C)ONC(=O)CSCC)NC(C(=O)NCC#C)(C)C c1(C(=O)CC)cccc(S(=O)(=O)N2CC3C(CO)C3C2)c1.N1(N)CCc2[nH]ccc2C1 Cc1nc2cnn(C)c2cc1C(N1CCC2(CCCC2NC(=O)C=CCO)C1)=O CCC(C(=O)N(C)Cc1cccc(C(F)(F)F)c1)C(C)O.C1(=O)CCNCCN1 c1(C(=O)NC(CC=C)CNC(C2CCOC2)=O)ccc2[nH]c(=O)cnc2c1 c1(OC)ccc(CC(=O)NC(C2CCN(C(c3ccc(C)s3)=O)C2)C)cc1F C#Cc1ccccc1CC(=O)N(CC(C)(C)NC(C1SC2C=CC1CC2)=O)C N1(C(C2CC(C)OC2)=O)CC2CCCC(NC(=O)C3=COCC3)C2C1 c1(C(N2CCCC(N(C(Cc3c(C)noc3Cl)=O)C)C2)=O)cccc(F)c1F c1(COC)nc(N2CCC(NC(c3ccc(C(=O)NC4CC4)[nH]3)=O)C2)cc(O)n1 C(=O)(C(CC1CCCC1)N1CCCC1c1cccs1)NCCCOC C1(C(N(C2CCN(C(C3(CC)CC3)=O)CC2)CC)=O)CCc2c[nH]nc2C1 C1(C(=O)NC2C(CNC(C3CN(C)C3)=O)CC2)COCC1(C)C N1(C(C2C3N(C(C4C(OCC)C4)=O)C(CC3)C2)=O)CCc2c(O)noc2C1 C1(NC(Cn2c(C)nnn2)=O)CCC2CC1CN2C(C1CC2(CCO1)CC2)=O C#CCC(O)C(=O)N1CCCC1C(N1CCC1C1CCCC1)=O c1(C(=O)NCC2C(NC(c3c(CC)nc[nH]3)=O)CC2)cn2ccc(CO)cc2n1 Cc1cn2cc(CC(=O)NCCCN(C(=O)CC3CCC3C3CC3)C)nc2s1 C=CCC(CC)C(=O)NC1CCC(F)(CNC(c2cc3n(n2)CCC3)=O)C1 N1(C(COCCCOC)=O)CC2CCC2(CNC(c2cccc(=S)n2O)=O)C1 C12(C(=O)NC(CC)CO)CCC(C(=O)NCc3cncs3)(CC1)CC2 C(CN=c1cc(NCC2CC(n3ccnc3)C2)nc[nH]1)c1cc(Br)ncc1 c1(C(=O)NC(C)CNC(=O)Cn2cc(N)cn2)ccc(Cl)nc1Cl CCCCCC(CC)C(=O)N1CCC(C2(NC(c3csc(CCC)n3)=O)CC2)C1 C1(C(=O)NC(C=C)C(F)(F)F)CN(C(c2cn(C)nc2C)=O)CC1(C)C C1(NC(c2cc(C)ncc2)=O)CC12CCN(C(c1cnc3n1CCCC3)=O)CC2 c1(CN(C(=O)NCC2(CO)COC2)CCc2ccccc2)ccc2nn[nH]c2c1 c1(-c2cn(C(C)C(=O)NCCSc3ccc(Cl)cn3)nn2)cc(F)c(F)cc1F N1(C(C(c2ccc(C)s2)C)=O)CCC2(CC1)CC2NC(=O)COc1ccncc1 C1(NC(CC=C)=O)CN(C(=O)COc2ccc(C(F)(F)F)nc2)C2(CCC2)C1 N1(C(c2c(C)scc2)=O)CCN(C(C2OCCOC2(C)C)=O)C(C(F)F)C1 C=CCCC(C(=O)NCC(=O)NCC=C)NC(=O)C(N1CCOC1=O)C CC(C)(C)CC(O)CNC(C1(NC(=O)CC2CC2)CCSC1)=O c1(C(=O)NC2C(OC)CN(C(c3ccc(O)cc3F)=O)C2)cc([N+](=O)[O-])c(C)s1 c1(OC)nc(C2=NOC(CC(=O)OC)C2)cc(CC)c1CC O=C(C1CCc2ccccc21)NCC1CN(C(c2ccn3c2CCCC3)=O)C1 c1(C(=O)OC)ccc2c(c1)CCCC2NC(C1C(C)(C)C(OC)C1(C)C)=O O=C(C1=CCCCCC1)NCCOCCCSCCOC1CCO1 c1(C(N(C2CCN(C(=O)CCC3CCCO3)C2)CC)=O)cn(CC)nc1C N1(C(c2ncn(C)c(=O)c2)=O)CC2CCC(NC(C3COC(=O)N3)=O)CC2C1 CC(C)CC(C(C)(C)C)N(C(C)C(c1ccccc1)O)Cc1cc(OC)c(Br)cc1I C(=O)(C(C)S(N)(=O)=O)NCC1(O)CC(CNC(Cc2cccc(C(C)C)c2)=O)C1 C(CCCCC(=O)NCCNc1ccccc1)C1C(C)C1.C1(CC2CC2)CC(=O)N1 c1(CCCC)cccc(C(C(=O)NC)N(CCC2(C)CCOC2)C)c1 Cn1cc(COC(C2CCc3c[nH]nc3C2)=O)c2ccccc12 c1(C(N(C2CN(C(CCC)=O)C2)C)=O)cnc2n1CCC2 c1(OC)cc(Oc2cncc(Br)c2)cc(C(=O)NC2CC2C(=O)NCCO)c1 N1(C(CCc2c(C)n(C)nc2)=O)CC23CCCC2(C1)CN(C(=O)CC(F)(F)F)C3 Cc1ccc2c(c1)CN(C(=O)CC1CCCN1C(c1csc(=N)[nH]1)=O)CC2 CN(C)NC(=O)CCC(=O)NC1(C2CCCN(C(=O)CCOC3CC3)C2)CC1 C1(NC(C2N(C)CCC2)=O)C2CN(C(c3cccc(NS(C)(=O)=O)c3)=O)CC12 c1(-n2cc(C(C)(C)NC(C(C)C)=O)nn2)ccc2cnccc2c1 C#CCC(C)(C)C(=O)NC1CC2(C1)CC(NC(=O)CC1CN3CCC1CC3)C2 Cc1ccc(C(=O)NC2CC(C)CN(C(=O)C(c3cn(C)nc3C)O)C2)cc1F N1(C(COCC=C)=O)CC(NC(c2ccc(-c3ccc(F)cc3)s2)=O)CC(O)C1 Cc1c(C(N2CC(N(C(=O)C=CCO)C)C3(CC3)C2)=O)cccc1C(F)(F)F C(=O)(CS(=O)(=O)N(C)C)NCC1C(NC(Cc2n(C)ncc2)=O)C1 N1(C(C(C)CO)=O)CCC2(C1)CN(C(=O)CCOC1CCOC1)C2 C1(OC)C(C)CN(C(=O)CCC(F)(F)Cn2cc(C(O)C3CC3)nn2)CC1C C(=O)(CCCCCc1nn[nH]n1)NC1(C)CCN(C(C)C)C1 C1(C(=O)NCCC(C)N(C(c2cn(C(C)C)nn2)=O)C)CCN(CCO)C(=O)C1 N1(C(C2CCC2)=O)CC(C2CC2)(C(=O)NCCc2csnn2)C1 C(=O)(C(C)C(=O)NCC1(NC(=O)C=C(C)Cc2ccc(Cl)cc2)CCOC1)OC c1(C(N2CCC(CNC(C3CCCC(OC)C3)=O)C2C)=O)ccnc2[nH]cnc12 c1(NC(C2N(C(=O)Nc3ccc(N(C)C)cc3)CC(O)C2)=O)nc2c(s1)CCC2 O=C(C1Cc2ccccc21)N1CCCC(F)(CNC(C2(Cl)CC2(F)F)=O)C1 c1(COC)nc(OC)cc(N2CC(O)(C(C)NC(c3c[nH]c(=O)cn3)=O)C2)n1 C=C(C)C(O)CC(=O)NCCN(C(=O)CNc1ccc(CC(N)=O)cc1)C c1(C(N2C(CNC(c3c(C)nc4sccn43)=O)CC2)=O)c(Cl)nc2ccccn12 c1(C(=O)NCCCC(O)C(=O)NC2CCCC(O)C2)ncn2ccccc12 N1(C(C(C)OCC2CCCO2)=O)CC2CCCC(NC(=O)C3=CCCC3)C2C1 C1(C(=O)NCCNC(N2CC(O)(SC(C)C)C2)=O)(C=O)CC12CC2.CCOC N1(C(CC2CC(C)C2)=O)CCN(C(c2ccnn2C(F)F)=O)CC1CF C(N=c1[nH]c(=NCC(CC)CCCC)c2sccc2[nH]1)c1n(CC)nnc1C C1(O)(CCNC(=O)Cn2cnccc2=O)CCCN(C(C2CCCS2)=O)C1 N1(C(C(CC(C)C)C)=O)CCC2CN(C(c3cccc4c3COC4)=O)CC2CC1 N1(C(C2CCN(C)C2)=O)CC(NC(c2csc(-c3nncn3C)n2)=O)C(O)C1 c1(C(=O)NC2CCN(C(=O)CCc3cnn[nH]3)C2)cc(Cl)cc2ccncc12 C1(CNC(C2CCC(CC)C2)=O)CN(C(C2(n3cccn3)CC2)=O)CC12CC2 N1(C(C2CCC(C(N)=O)O2)=O)CC2CC2(CNC(C2CC(F)(F)C2)=O)C1 CCC(C)(C)C(=O)NCC(C(=O)NC1CC=C(C)CC1)N(C)C C(=O)(C(C)CS(=O)(=O)c1ccc(Br)cc1)NCc1cc(OC)c(OC(C)=O)cc1 c1(OC)cc(NC(C2CCN(CC3CC4CCC3O4)C2)=O)cnn1 N1(C(CC(CCC)C)=O)CCC2CCN(C(=O)Cn3ncnn3)CC2C1 C1(CNC(C2N(C(C(C=CC)O)=O)CC2)=O)CN(C)CCN1C N1(C(CC2C(C)C2)=O)CC2CCCC(NC(c3ncccc3O)=O)C2C1 C1(NC(C(C)Oc2cccnc2)=O)CCC2CN(C(c3cnoc3)=O)CCC2C1 C1(C(N2CCC(C)(NC(=O)CC3CC34CC4)C2)=O)(OC)CCOCC1 c1(C(N2CC(O)(C(C)NC(C3CCCOC3)=O)C2)=O)cc([N+](=O)[O-])c(O)cc1N N1(C(C(C2CN(C(C3(C(C)C)COC3)=O)C2)N(C)C)=O)CC(O)(C2CCC2)C1 CN1N=C(CC(=O)N2CCOCC(NC(C3(n4cccn4)CCC3)=O)C2)CC1=O C1(C(NOCCC2CC(=C)C2)=O)CC(COC)CCO1.n1(CC(=O)N)cc(C#N)cn1 c1(C(=O)NCC(C)(CO)NC(C(C=CCCC)O)=O)ccc2c(c1)COCC2 Cc1cc(C(F)(F)F)nc(N2CC3C(NC(c4ccc(F)cc4Cl)=O)C3C2)n1 Nc1c(Cl)cc(C(=O)NCC2CC(O)CN2C(=O)CCOCC2CC2)c(O)c1Cl C1(C(=O)NCC(O)CNC(c2csc(O)n2)=O)(CC)CCCC1O Cc1noc(C(CO)NC(=O)CCNC(=O)C(C)Cn2cccn2)n1 c1(C(N2CC(O)(CCNC(c3cc(F)ccc3F)=O)C2)=O)cc(F)c(O)c(F)c1 C1(C(C)C)CCC(NC(C2CC23CC(OC(C)(C)C)C3)=O)CC1 CCN=C(NCC1CCCC(SCC)C1)N1CCC(CC)C1 c1(CC(C)NC(=O)NC(C2CCCO2)CC)ccccc1Cl c1(N2CC(C)C(NC(c3cc(Cl)cn3C)=O)CC2)ncc2c(ncn2C)n1 CC1CC(C(=O)NC(C)(C)CNC(=O)COC2CCCCCC2)CC(C)C1 Cc1cc(Cl)c([N+](=O)[O-])cc1C(N1CCC(CC(=O)NC2CC2(F)F)C1)=O C#CCCCCC(=O)NC(CCC)CCCNC(c1nc(SC)ncc1N)=O C(CCCCC(=O)N1C(C(=O)NOCC2CC2)CCC1C)SC c1(OCC(=O)N(C(CCNC(C=CC(=C)C)=O)C)C)ccc2ccc(=O)oc2c1 C1(C(=O)NC(C)(CNC(C2(CO)COC2)=O)C2CC2)SCCCS1 C(C1=NOC2CCCC12)NCC1CCS(=O)(=O)C1 C#CCC(C)C(=O)NC(C)CNC(C12CC(N3CCN(C)CC3)(C1)C2)=O c1(C(N2CC(CNC(C=NOC)=O)C(C)(C)C2)=O)cc(N)c(F)cc1F C1(CNC(C(=C2CN(C(C3CC(OCC)C3)=O)C2)F)=O)CC2CCCCN2C1 C1(NC(C2(OC)CCCSC2)=O)CCN(C(=O)CC(C)(C)N(C)C)CC1C CC1CCC(=CC(=O)N(C2CC2)CC2(CO)CC2C(F)(F)F)C1 C1(C(N2C(c3onc(COC)n3)CCC2)=O)CCCN(Cc2ccc(C#N)s2)C1 C1(C(=O)NCCCOCCNC(c2c(CCC)onc2C)=O)CCC(C)NC1=O c1(OC)ccc(CCC(=O)N2CC(CC(C)NC(=O)C3=CCCC3)C2)c(F)c1 C12(NC(CCC=C)=O)CCCC1CN(C(c1cccc(F)c1C)=O)C2 C12(CNC(c3cc(O)cs3)=O)CC1CN(C(C1CCO1)=O)C2 C1(NC(N2CC(C)(OCC)C2)=O)C2Cc3c(Br)cccc3C12 C1(NC(CC2C(CC)C2(F)F)=O)CC2(CCN(C(c3csnn3)=O)CC2)C1 Cc1cccn2cc(C(=O)NCC3CCC3NC(C3(CF)CCC3)=O)nc12 CCC(C(=O)NC(CC(=O)N(C1CCCC1(C)O)C)C1CC1)C(F)(F)F C(CC(C)C(C)(C)C)NC(C#C)CCC(=O)OCc1ccccc1 C(CCC(=O)N1CCC1(C)C(C)C)(C(C)C)NC(c1c(CC)oc(C)c1)=O C1(C(=O)NC(C2CCCN2C(C2CSC2)=O)C)CCC2(CC1)NC(=O)N(C)C2=O C1(NC(C(CCC)NC(CC=C=C)=O)=O)CCOC12CCCC2 N1(C(c2c(N)ccc(Cl)c2)=O)CC2(CCCC2NC(C2CC2F)=O)C1 CC1CC(NC(c2cccc(=O)n2C)=O)CCN1C(c1cc(Cl)cnc1O)=O C12(CNC(c3n(C(C)C)ccc3)=O)CCC(C1)N(C(=O)Cc1sc(O)nc1O)C2 Cc1cc2nc(Cl)nc(N(CC(C)NC(=O)CN3CCOCC3)C)c2s1 C1(C(=O)Nc2c(C#N)cncc2)CCC2(CN(C(c3sc(Cl)nc3Cl)=O)C2)O1 C1(NC(=O)Nc2ccc(C)cc2I)CCC2(CC1)CN(S(=O)(=O)CCCl)C2 c1(OCC2CC(NC(C3(OCC)CCCCC3)=O)C2)ncnc(OC)c1F C1(C(=O)NCC23CC(NC(C(CC)N(C)C)=O)(C2)C3)CC2CCC1O2 C1(NC(=O)CCc2ccco2)CCCCC1NC(C1CCC1c1ccccc1)=O C1(C(N(CCCNC(C(C)C#N)=O)C)=O)CCC2(CCCO2)CC1 CC1(C)NC(=O)CC1C(N1CC(C(=O)NCc2cc[nH]n2)C2(CC2)C1)=O C12(NC(CSCC(N)=O)=O)CCCC(CN(C(=O)CNC(=O)NC3CC3)C1)C2 N1(C(CSCC(C)C)=O)CCC(F)(CNC(=O)C(C)NC=O)C1 CCCC(C(=O)OC)C(=O)N(CCNC(c1cnccc1C(F)(F)F)=O)C1CC1 C(=O)(C(CC)(CC)CO)NC(CCCNC(c1ccc(C2(COC)CC2)o1)=O)C c1(-c2ccc(C(C)O)cc2)cc(=O)n(C)c(O)n1 N1(C(C)C(=O)NCCN(C(c2ccccc2)=O)CC2CCCO2)CCCCCC1 N1(C(c2c(CC)n[nH]c2)=O)CC2CC1CN2C(C1CCC(COC)C1)=O CCC(CCc1ccccc1)NC1CCC(C)C1 Cc1ccc(NC(=O)CN2CCN(C(=O)COC3(C)CCOCC3)CC2)c(O)c1 C1(F)(C(N2CC(F)(CC(=O)NC3(c4c(C)cno4)CC3)C2)=O)CC=CCC1 c1(C(=O)NC2C(CC(C)(C)C)CCC2)cc(Br)cc(S(C)(=O)=O)c1F C1(NC(c2c(C)cnn2C(C)C)=O)CC(C2CCN(C(=O)C3=CCSC3)C2)C1 O=C(CC(F)(F)F)NC1CC12CC(NC(=O)C1=CCC1)C2.C1CC(=O)N1 c1(COC)ccc(Cl)c(CNC(=O)CC2CCC(O)C2)c1 c1(OC)cnc(C(N2CCCCC2CNC(=O)CCCCSC)=O)c(F)c1 N(C(=NCC(C)c1cccs1)NC1CCC1)Cc1cc(OC)c(F)cc1 Cc1cc(=NCCc2cn3c(n2)SCC3)[nH]c(=NCc2nc(=O)n(C)[nH]2)[nH]1 CCCC(C(=O)NC12CC(CNC(c3ccc(C(C)=O)o3)=O)(C1)OC2C)C(C)C C1(CNC(C(C)OCC)=O)(NC(c2ncc(Br)cc2F)=O)CCCCCC1 C1(C(=O)NCC2(C)CCCN(C(C(C)C3CCC3)=O)C2)COc2ccccc2O1 N1(C(C(CC)OC)=O)CCOCCC1C(=O)Nc1cnc(OC)cc1C C#CCC(CC(=O)NC1CC(O)CCN1C(=O)CCC1CC(OC)C1)OC c1(C(CC2CCCO2)N(CC)CC)cc(C)ccc1F.c1(CCCN)ccc(O)cn1 CC(C)C(C)(O)C(=O)NC1CC2CN(C(=O)C(=O)NCC(F)F)CC12 C1(C(=O)NC(C2CN(C(C(C)NC(C)(C)C)=O)C2)C)CSc2ccccc2O1 c1(C(=O)NCC(CNC(c2scc(OC)c2)=O)OC)cc(SC)c(C)o1 C(=O)(CC(C(F)(F)F)n1cccn1)NC1CCN(C(C2CC(SC)C2)=O)CC1F N1(C(C=C(C)C2CC2)=O)CCOC(CNC(=O)CN2CC(C)C2)C1 N1(C(CC(C(=O)OC)C)=O)CCCC(C2(NC(=O)C(CO)N(C)C)CC2)C1 Cc1cn(CC(=O)NC2CCCC(C(=O)NCC3COC(C)(C)C3)C2)c(=O)nc1O Cc1sc(C(N2CCCCC(C)C2)C(=O)NCCCF)c(C)c1C CCC(C)(C)C(C)CC(=O)N1CC(O)(CNC(C2CC3C=CC2CCC3)=O)C1 c1(CC)cc(C(=O)N(C2CCN(Cc3cn(CC(=O)NC(C)C)nn3)C2)C)ns1 c1(C2(C(N(C3CCN(C(C(CC)N(C)C)=O)C3)CC)=O)CC2)ncccc1F N1(CC(=O)NCC2(O)CN(C(C3C(C)(C)COCC3)=O)C2)CCCCC(O)C1=O Cc1cc(N2CCC(c3nc(O)n[nH]3)CC2)nc(N2CCC(CS(N)(=O)=O)C2)n1 S(=O)(=O)(c1ccc(F)c(Br)c1)Nc1cnn2c1CN(C(C1(C)CCC1)=O)CC2 c1(C(=O)NCC2CCC(NC(CCc3c(C)noc3)=O)C2)ccc(N)c(O)c1 C(=O)(C1=COCCC1)N(CC(CNC(C=Cc1ccc(CC)o1)=O)(C)C)CC c1(C(C(=O)O)NC(C(c2ccccc2)N(C(C)=O)C)=O)cccc(C(F)(F)F)c1 C12(NC(C3CC(O)(CC#C)C3)=O)CCCC1N(C(=O)C(c1ccccc1)F)CC2 C1(C)(CNC(c2c(C)noc2C)=O)COCCN(C(C2CCCCN2N=O)=O)C1 C1(CNC(C(CC)n2cncn2)=O)CCCN(C(=O)CCCn2cncn2)CC1 N1(C(C(OC)OC)=O)CCC(NC(C2CCCCN(C)C2=O)=O)C12CCC2 c1(C(=O)NC2CC(F)(CNC(CS(C)(=O)=O)=O)C2)ccc2cnnc(O)c2c1 C#CC(C(C)(C)C)NC(C1CC12CC(NC(=O)CCc1cncs1)C2)=O C1(C(=O)NCCCC(C)NC(=O)Cc2ccon2)CC1C1CCOCC1 C#Cc1cn(C)nc1C(=O)NC1(C)CCCN(C(=O)Cc2csc(C(C)C)n2)C1 Cc1nn(C)c(Cl)c1-c1cn(-c2cccc(CNC(C3(C)CC3(Cl)Cl)=O)c2)nn1 C(CC(C(=O)NC1CN(C(=O)CC2COCC2O)CC1C)NC=O)SC CC1CCC(NC(C2CC(C)(F)C2)=O)CN1C(c1csc([N+](=O)[O-])c1)=O Cn1nc(C(N2CC3CN(C(=O)CC(C)(C)C#N)CC3(C)C2)=O)c2ccccc12 C1(C)(C(=O)OCC(C)C(=O)Nc2ccccc2)CCCOC1 C1(CCNC(=O)CNC(=O)N)CCCCC1.CC(C)(C)OC(=O)NCC1CC1C S(=O)(=O)(c1cccnc1NCC1(CO)CCC(=O)N1)NC(C)CC1CCC1 C1(CC)CC(C(N2CC3(CCC3O)C2)=O)CCN1C(=O)CCC1(C)CC1 c1(NC(C2CC(NCc3ccc(C#N)c(Cl)c3)C2)=O)cc(Br)cc([N+](=O)[O-])c1 C12(CNC(C3(CC#C)CC3)=O)CCC(CC1)N2C(=O)CCC(C)n1cccn1 Cc1coc(C)c1C(=O)NCCN(C(C1CCC2CC12)=O)CC1CC1 c1(C(N2C(C)(CNC(c3cccc(CO)c3)=O)CCC2)=O)cc(N)cc(N)c1 c1(C(=O)NC(CC)CNC(=O)C=C(C)C2CC2)ccc2c(c1)OC(C)(C)CS2 N1(C(c2c(SCC=C)cccc2)=O)CCC2(CC1)CN(C(=O)CCC)CCO2 N1(C(C(CSC)OC)=O)CCC(N2CCC(NC(=O)COC(F)(F)F)CC2)CC1 c1(C(N2C(CNC(C3CCCSC3)=O)CC(OC)C2)=O)cnn2cc[nH]c(=O)c12 CCC(C(=O)NC1(C)CN(C(=O)COCC2CCCC2)C1)n1ccc(C2CC2)n1 C(=O)(CCC(N)=O)N(C1CCN(C(c2ncn(C)n2)=O)C1)N1CCCCC1 C(=O)(CC(C)(C)C(C)(F)F)NCC1CN(C(C(C)OCCN(C)C)=O)CC1C c1(NC(=O)NC(C)CC(=O)OCC(F)(F)F)ccc(C(C)O)cc1 C1(NC(Cc2c(C)con2)=O)C2CC3C(C2)C13C(=O)NCCC(C)C(F)(F)F N12CCCC(C1)N(C)C2=O.c1(C(=O)NC)nc(COC2(C)CCCC2)cs1 C(N=c1[nH]c(C)ncc1F)C1C(NC(C(n2cc(C)cn2)CC)=O)COC1 c1(C(N2C3CN(C(CCc4scc(C)n4)=O)CC2C3)=O)cccc2occc12 C1(C(C)(C)NC(CC2C(OC)C2)=O)CCN(C(C2(C3CCCO3)CCC2)=O)CC1 c1(C(N2C(CC)CN(C(=O)C(C)N(C)C)CC2)=O)cc(=O)c2cc(F)ccc2o1 N1(C(C(C2(OC)CCCCC2)(F)F)=O)CC2CC(NC(=O)CC(C)C(C)C)C1C2 c1(SC)nc(C)c(NC(=O)Cc2ncccc2C(F)(F)F)s1 Cc1cnn2cc(C(=O)NCC3CCCN(C(=O)C=Cc4cscn4)C3)cnc12 C1(O)(CNC(C2C(=O)NCC2)=O)CCN(C(=O)COC(F)(F)C(F)(F)F)C1 c1(C(N2CCC(OCC(C)C)C2)C(=O)NC(CC)C)ccc(S(N)(=O)=O)s1 C(=O)(CCS(C)=O)NCC(CNC(c1ccc(COC)s1)=O)O OC1Cc2ccccc2CN(CCc2ccsc2Br)C1 CN1CCN(C(C2CCCCCC2)=O)C(CNC(C2CC(n3cnnc3)C2)=O)C1 CC1(C)OC2CC(C(N3CC4CN(C(C5CC5(C)Br)=O)CC4C3)=O)CC2O1 c1(C(=O)NC2CN(C(CCSCC(N)=O)=O)CC2O)cc(F)cc2ccccc12 CCCCC(CNC(=O)C(F)=C1CCC1)NC(=O)CSc1nccn1C N1(C(c2cncc(OCC)n2)=O)CCC2(CCCN(C(=O)CNC(=O)NC)C2)C1 c1(CC)nnc2n1CCN(C(=O)NC(c1c(Cl)ccc(F)c1Cl)C)C2 C1(C(=O)NCCN(CCOC)C(C2CC2CC(C)C)=O)(CC)CCCC1 N1(CC(=O)NCCCN(C(c2nc(C(C)C)sc2)=O)C2CC2)CCC(C)CC1 Cn1ncc2ncnc(N3CC4(CN(C(=O)C#CC5(C)CCCO5)C4)C3)c12 C=C(C)CCC(=O)NCCOCCCN(C(=O)Cc1cnoc1)C.C(CO)O c1(C2(NC(c3c(C)coc3)=O)CC2)ccc(C(=O)N(C2CCCCCC2)C)cc1 N12CCC(COC)(C1)CNC(=O)C2(F)F.C1(CCOC)CC1C=O.C1CC1 CONC(=O)C(=O)NC(CCSC)C(=O)N(C)CC1COCCO1 N1(C(c2cnc(C(C)O)s2)=O)CCSCC1CCNC(c1cc(F)c[nH]1)=O CCCCCCCCC(F)C(=O)NC1CC2CC1N(C(=O)CNC(=O)CCC)C2 c1(C(N2CC(O)(CN(C(c3cn(C(C)C)nc3)=O)C)C2)=O)c[nH]c2nccc-2c1 C1(C(C)O)CN(c2nnnn2CC(c2ccccc2)C2CC2)CCO1 C(=O)(C1=NOC(C)C1C)NCC1C(C)C1.c1(C(NOC(C)C)=O)ccn(C2CC2)n1 c1(C(C)Nc2cc(N3CCCC(N4CCC4)C3)ncn2)cc(Cl)ccc1F C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)N1CCCC(NC(c2n[nH]cc2Cl)=O)C1 N1(C(CSCC=C)=O)CCN(C(c2csc(C(F)F)n2)=O)C(CCCC)C1 C(C(C)(C)C(=O)NCC(c1cnn(C)c1)C)N(C(c1n(CC)ncc1)=O)C c1(C(N2CCN(CC(F)F)CC2)C(=O)NCCCOC)ccnc(P(C)(C)=O)c1 C1(N(C)C(=O)O)CCc2n[nH]cc2N1CS.N1(CCCN(CC(C)C)C)CCCCC1 Cc1scc(C(N2CCN(C3CN(C(=O)Cc4cnc(C5CC5)[nH]4)C3)CC2)=O)c1N C(C(O)CC(=O)NOC1CC1)NC(=O)CC1CCCOCC1 C(=O)(C(CCC(N)=O)=CCC)NCC(CC=C)NC(=O)C(C(C)O)NC(C)=O C1(NC(c2c(C)n[nH]c2)=O)CCC2CN(C(c3ccncn3)=O)CCC2C1 C1(NC(=O)CC2CC(C(F)F)C2)CN(C(=O)C=CC2CCCO2)CC1C1CC1 c1(C(N(C(CNC(=O)C(c2cncn2C)O)C2CC2)C)=O)ccncc1F C=C(C)CCCC(=O)N1CCC(OCCNC(=O)CC2CCCOCC2)C1 C(=O)(C(O)CC(N)=O)N1CCC(C(C)(C)N)CC1.c1(C(=O)OC)cc(C2(C)CC2)[nH]n1 Cc1ccc(C(N)=O)cc1C(=O)NC1CC1NC(=O)CCc1cccc(O)n1 N1(C(CC(CC)CC)=O)CC2CCC(CNC(=O)Cc3sccc3C)C2C1 C1(n2cccn2)(C(=O)NCCCN(C(CSCCOC)=O)CCO)CCC1 N1(C(c2c(C)ccs2)=O)CC(NC(c2cc(F)cc(F)c2)=O)CC12CCC2 Cc1cc(S(N)(=O)=O)sc1C(=O)NC1C2CN(C(=O)C#CC3CCCCC3)CC12 Cc1cccc(C(=O)NCC2CC2CNC(=O)Cn2ccc(C3CC3)n2)c1F N1(C(C(C2CC(CC(=O)NC3CC=CCC3)C2)F)=O)CC(C2CCCC2)C1 c1(C(N(CC(CNC(CC(C)C2CC2)=O)O)C)=O)ccn2c1CSCC2 C1(NC(CCOC(C)=O)=O)CC(F)(F)CC1NC(=O)CCC1CCCN(C)C1 C=CC(C)(CCOC)C(=O)N1CC2(C(N3CC(S(C)=O)C3)=O)CC1CO2 c1(CC)nn(C)cc1CNC(=O)CNC(=O)CNC(=O)CC1CCN(CC)CC1 c1(C(N2CCCCC2CO)=O)cc(-c2ccc(OC(F)F)cc2)cc2c[nH]nc12 C1(C(N(C)CC2N(C(C3CCC(C)C3)=O)CCC2)=O)CCC(O)CC1 C12(NC(C3CN(C)C3)=O)CCC(CNC(c3occc3Cl)=O)(C1)OC2 N1(C(CC2CCN(C(c3n(CCC)ncc3)=O)C2)=O)CCSC(C)(C)C1 C1(C(=O)OC)CC(n2cc(C)nn2)CN1CCC(C)C.C1(C(=O)N)CC(C)=NO1 C1(NC(CCN(C)CC)=O)CCN(C(c2nc(C)oc2C)=O)CC1CO N1(C(CCC=C=C)=O)CCN(C)CC1CN(C(c1ccnn1C1CC1)=O)CC N1(C(c2c(CC)[nH]cc2)=O)CC2CCC(C1)C(NC(=O)CCn1ccnc1)C2 c1(C(=O)NC(CCN(C(C2(CCC)CC2)=O)C)C)cc(Br)cc(F)c1F C1(CN(C(=O)CCC2CC2)CC)CCCCN(C(=O)Cc2ccn(CCF)n2)C1 C1CN=C2N=c3c(cnn3C)=C(N2)NC12CCCC2.C1(COC)CCN(C)CC1 c1(N(C2CC3CNC2C3)C(c2cc(O)cc(Br)c2)=O)nc(O)c2nc[nH]c2n1 c1(C(=O)NC2CC(NC(=O)C(F)C3CCOC3)C2)cc(O)ccc1[N+](=O)[O-] c1(C(=O)NC2C(C)(C)CN(C(C3CCCOCC3)=O)C2)csc2c(O)ccnc12 C1(F)(CNC(C(C(C)C)NC=O)=O)COCCN(C(C2CC2(F)F)=O)C1 c1(CC(=O)N(C(C)CNC(=O)C(C)n2cncn2)C)nsc2ccccc12 C(=O)(CCCCCCS(N)(=O)=O)N(CCCC=C)C.c12cn(nn1)CC2 Cc1cc(C(=O)N(CC(O)CNC(=O)CCc2nnc(C3CCCC3)o2)C)sn1 C#Cc1cn(C)nc1C(=O)NCC(C)(C)CC1(NC(C2CCCCC2C)=O)CC1 C(=O)(CC(O)CC(C)(C)C)N1C2C(NC(Cc3c(C)ncc(Cl)c3)=O)C(C2)C1 c1(C(N2CC(C(C)NC(COCCC(C)C)=O)C2)=O)cocc1C(N)=O N1(C(CCNS(CC)(=O)=O)=O)CCCC1C1(O)CN(C(c2ccc[nH]2)=O)C1 C(=O)(CCCC(=O)N(C)C)N1C(CCC(N2C(C)CCCC2)=O)CCC1 c1(C(N(C(C)CCNC(c2cc3occc3s2)=O)C)=O)cnc2ncnn2c1N N1(CCNC(C2NC(=O)OC2)=O)CCN(C(C2CC(CF)C2)=O)CC12CCC2 C12(CNC(C3C(C)OCCO3)=O)CCCC1CCN2C(c1cc2ccsc2s1)=O c1(OC)cc(C)c(C(N2CC=C(CNC(C3(C(F)F)CC3)=O)CC2)=O)cn1 c1(C(N(C)CC2CCN(C(C(CC)O)=O)C2)=O)ccc(S(=O)(=O)NC(C)C)cc1 C1(C(N2CCC(O)(C(=O)NC(C)(C)CN3CCCC3)C2)=O)CC=CC(O)C1 C=CCCC(C(=O)N1CC(O)(CC(C)C)C1)NC(c1c[nH]c(=NC)s1)=O C(C(CC(C)C)C(=O)N1CC2(CC(NC(C3CC(C)OC(C)C3)=O)C2)C1)OC c1(CN(CCNC(CC=CC=C)=O)C(c2cnc(C(C)C)[nH]2)=O)ccc(Cl)nc1 n1(CC(=O)NCCC2CN(C(c3c(CC)ocn3)=O)CC2C)ccc(C)cc1=O c1(C(=O)NCC(CNC(=O)CC2CC2(C)C)OC)ccc(Br)c(N)c1 C1(C(=O)NCC2C(CNC(c3csnn3)=O)C2)Cc2c[nH]cc2S1(=O)=O C#CC1(C(N2CC3(CC3)C2)=O)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 CS(=O)c1ccc(C(c2nnnn2C2CC2)NC(c2ccc(Cl)cc2)C2CC2)cc1 Cc1nn(C)c(C)c1CNC(C1CCCN1C(=O)CCCC1CCCC1)=O c1(OC)ccc(C(C)NC(=O)NC(C)C(c2cccc(F)c2)O)c(C)c1 c1(C(=O)NCC#CCNC(C2(O)CC(C)(C)C2)=O)cnc2[nH]ncc2c1 c1(C(N2C3CN(C(c4csc(Cl)n4)=O)CC2CC3)=O)ccc2c(c1)CCNC2=O Cc1cc(C(=O)NC2CCCCC2NC(C2CC(C)OC2C)=O)c(O)c(C)c1 N1(C(COC)=O)CCC2OCCN(C(=O)CN3CCCCC(O)C3=O)C2C1 c1(C(=O)NCC(C(=O)NCC2OCCN(CC)C2)O)ccc(F)c(F)c1 C(=O)(CC1OCc2ccccc21)N(C1CCN(C(=O)CC2(CO)CC2)C1)CC C1(C(=O)NCC(=O)NCC(=O)NC23CCN(CC)CC2C3)C2(CCC2)C12CCC2 c1(C(N2CCCC(N(C)C(c3scc(Cl)c3Cl)=O)C2)=O)c(C#N)cnn1C N1(C(CCC)C(=O)Nc2ccc(OC)cc2C)CCc2cccc(Br)c2C1 Cc1cc(C)c(C(=O)NCC2CN(C(C3(C)CC=CCC3)=O)CCO2)cc1C C1(C(c2cc(F)ccc2F)c2onc(C3(C)CCCC3)n2)CCCCC(=O)N1 c1(C(=O)NCCCNC(c2ccc(SCC)o2)=O)cc(OC)c(OC)c(N)c1 c1(OC)cc(C(N2CC(NC(=O)C=C3CCC(C)C3)C(C)(C)C2)=O)c(O)c(Cl)c1 c12c(noc1C)NC(=O)C(COC)NC2=O.C(=O)(CC1(CSC)CC1)NC C1(NC(c2c(O)ccc(OC)c2)=O)CC2(CCCCN2C(=O)C2CC2)C1 C1(C)(C(N2C(CCNC(C(CC)NC(C)=O)=O)CCC2)=O)CCN(C)C1=O C(CCCCC(=O)NC1(CC(N)=O)CCN(C(C2CCC2(OC)OC)=O)CC1)OC N1(C(=O)CCc2ccccc2)CCC2(CCCN(C(C3(F)CCOC3)=O)C2)C1 N1(C(CN2CC(CC)C2)=O)CC(CNC(=O)C(C)(C)CO)C(F)(F)C1 c1(C(N(C)CC2(O)CN(C(=O)C(C)(C)NS(C)(=O)=O)C2)=O)cc2cccnc2[nH]1 c1(CN(C(=O)CN2CC3CCCCC3(CO)C2)CC)cccc2ncccc12 Cc1cc(C(F)(F)F)cc(C(N2CC(NC(=O)CC3CCOC3)CC(F)C2)=O)n1 C(=O)(NN1CCCC1C(=O)NCc1c(C)cnn1C)c1c(C)csn1 C1(CN(C(=O)CCc2ccc(C)cc2)CC)CCN(C(C2COC(=O)O2)=O)CC1 C(=O)(C(C)(C)CCSC)NCC(CNC(c1ccc(CC(=O)NC)cc1)=O)O CCC(C)(CO)C(=O)NCc1cn(C2CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)nn1 N1(C(C(CNC(C(CCC)F)=O)N(C)C)=O)CCN(CC(N)=O)C(=O)C1 C1(N(C(C2CN(C(C)C)C(=O)C2)=O)C)CCC2CN(C(=O)CNS(C)(=O)=O)CC12 C1(C(=O)NC2CN(C(c3cc(C)no3)=O)CC2C(F)F)CN2CCC1CC2 C1(CNC(C(C)(C)n2cc(Cl)cn2)=O)COCCN1C(=O)CC1CCC(O)C1 S(=O)(=O)(CC(=O)NCCCC(C)NC(c1csc(-c2ccco2)n1)=O)NC(C)(C)C C1(NC(C(=O)NCC)=O)CC12CCN(C(c1c(F)cc(C)cc1F)=O)CC2 c1(CC)cc(OC)c(OC)c(CC(=O)NCC2CCN(Cc3ccsc3Br)C2)c1 N1(C(C(C)OC(C)C)=O)CCOCC1C(=O)NCCCCC1CC1 C1(C(N2C(CNC(c3ccnc(O)c3)=O)CC(F)(F)C2)=O)CCc2cncn2C1 CC1CCSC1C(N1CC(F)(CNC(=O)CCc2ncc[nH]2)C1)=O c1(CC)oc(C)cc1C(=O)NCCC(C)N(C)C(c1csc(=NC)[nH]1)=O C(=O)(C(C)(C)CNC(=O)CC1CC=CCC1)N(C(C)C)C C(=O)(C1COc2ccc(Cl)cc21)NCCC(C)NC(c1cn(CCF)nn1)=O C1(S(N)(=O)=O)(NC(C(=O)NC(c2cn(-c3c(C)c[nH]n3)nn2)C2CC2)=O)CC1 N1(CC)CCC(CN(C2CC2)Cc2ccccc2)C1.C1(C2CCC2)CNC(=O)N1 c1(C(=O)NCCN(C(C(C2CCCCC2)OC)=O)C2CCCC2)ccc(F)cc1F N1(C(C2CCCN(C(c3c(C)csn3)=O)CC2)=O)CCCC2(CC1)CC2 C=CCC(C)C(=O)N1CCCC1C(=O)NC1COCC1N(C)C C1(OC)CC(C(=O)NC2CC2NC(c2csnc2C)=O)N(S(C)(=O)=O)C1 O=C(CC1OC(=O)c2ccccc21)NC12CCCC1CN(C(C1(O)CCC1)=O)C2 N1(C(C2(SC)CC2)=O)CCC2C(C(=O)NC(CC#N)C3CC3)C2C1 N1(C(c2ccc(COC)[nH]2)=O)CCC2(CCCN2C(C23CC(C2)C3)=O)CC1 N1(CCCCC(C)C)CCC2(CC1)COC(CNC(=O)C(C)(C)C1CCCO1)C2 C1(C(C)NC(COCCCCC)=O)CCN(C(c2cc(C(C)(C)C)no2)=O)C1 C1(C(C)NC(=O)Cc2cnsc2)CCN(C(c2oc(C3CCC3)nc2C)=O)CC1 c1(C(N(CCNC(c2c(C)ncnc2)=O)C)=O)cccc(F)c1C(F)(F)F CN(C)NC(=O)CCC(=O)N1CCCC(NC(c2cnn3c2C(C)CCC3)=O)C1 C(=O)(C(O)CC[S+](C)C)NC1(CC)CCN(C(C2CC3(CCOC3)C2)=O)CC1 c1(C(=O)NC(c2ccccn2)C)cn2c(n1)CN(C(c1cc[n+]([O-])cc1)=O)CC2 N1(C(=O)CN(C2COC2)C(c2ccc(CO)cc2)=O)CCCC(CC2CC2)C1 CCCC(CC1CCCC1)C(=O)NCC1CCC(NC(C2CCN(C)C2)=O)CC1 C1(COC(C)=O)CCN(C(C2(C(C)N(C(=O)C(F)C3CCCC3)C3CC3)CC2)=O)C1 CC1(C(=O)NCc2ccccc2CNC(=O)CN2CC(=O)NC2=O)CCCCO1 N1(CCOC)CCC(CNC(=O)CC2(NC(C3CCN3C(C)C)=O)CC2)C1 C12CC=CC(C1)NC(=O)C2.c1(C2(C(C(C)O)C)CC2)nc(-c2ccccc2)n[nH]1 C1(NC(C2CC(OC)C2)=O)CC(C)(C(=O)NCCC2(O)CCCC2)C1 CN1CCOC(C(=O)NC2CCC23CN(C(C2CC=CC2)=O)C3)C1=O N#Cc1nc(=NCC2CC(CNC(c3cc4ccc(Cl)cc4[nH]3)=O)CO2)cc[nH]1 C(CCC(=O)NCC(CO)C(C)C)(C(C)C)NC(c1cc(C)nnc1C)=O CCC(CNC(=O)C(F)(F)Cc1ccccc1)(CC)NC(c1cncnc1C)=O c1(C(=O)NCC2C=CCN2C(c2cnc(S)[nH]2)=O)cc2nc(=O)ccn2[nH]1 c1(C(N(C2(C#N)CC2)C)=O)cnc2cc(Br)ccn12 C(=O)(C1CCc2cccc(F)c21)NC1C(NC(CCSCCCC)=O)CCCC1 O=C(CS(=O)(=O)Cc1cccs1)NCC1CC(NC(=O)CCC2CC2)C1 N1(C(c2cnn(C(C)C)c2Cl)=O)CC2CCN(C(C3CCC(=O)N3C)=O)C2C1 C1(C(=O)NC(C(=O)N2CC(CC34CC(C3)C4)C2)C2CC2)CC2(C1)CC21CC1 C1(NC(C2CCC(=C)CC2)=O)CCN(C(c2cc(F)ccc2C)=O)CC1C(C)C C1(NCC)CCCC(N=c2[nH]c3c(c(=NCC4(C)CC4)[nH]2)CSC3)C1 c1(NCC(C#C)OCC)ncnc2c1ccn2C1CC1 c1(OC)ccc(-c2cn(CCN(C(C3CC(F)(F)CS3)=O)C3CC3)nn2)cc1Cl c1(C(N2CCN(C(N)=O)C3C2COC3)=O)cc(C2CC2)nc2ccc(Cl)cc12 c1(C(N2CCCC(NC(C3C(C)(C)C3)=O)(CO)C2)=O)csc2ncnc(O)c12 CC1(C)CCCC(C(=O)NCc2csc(C(=O)NCC3CCCOC3)c2)C1 C(C1CCCN1C)=CC(=O)NCC1CCC(NC(C(C)OCC2CC2)=O)C1 C(=O)(C(C)(O)C(C)C)N1CC(Cc2c(C)cc(-c3cn(CCOC)nn3)o2)C1 CC1(CCNC(=O)CCC2CC(NC(c3cccnn3)=O)C2)CCOC1 Cn1ccc(C(=O)NCC(O)CNC(c2ccn(CCO)c(=O)c2)=O)c(O)c1=O n1(CC(=O)NC2C(NC(c3ccc(C)c(Cl)c3)=O)C2)ccc2ccccc2c1=O c1(C(=O)NCC2CN(C(C(C=CCCC)O)=O)C2)cc(F)ccc1Cl C(=O)(C(C(C)(C)C)N(C)C)NCc1cnn(C)c1C(=O)NCC(C1(C)CCC1)O C1(C(N(C)CC2CN(C(=O)C3=COCCO3)CCO2)=O)CCn2nncc2C1 c1(C(N(C2CCN(C(C3C(C)C3)=O)CC23CC3)C)=O)ccc(Cl)c2ccccc12 c1(OC(CCN(CC(F)C(=O)OC)CCCCC)=O)ccc(C)cc1C N1(C(C2N(CC)CCOC2)=O)CCC(CNC(c2conc2C(C)C)=O)C(O)C1 C1(C(=O)NC2(CNC(C(CC)O)=O)CCOCC2)CS(=O)(=O)CC(=O)N1 N1(C(CSC)=O)CCOC2(CCN(C(=O)Cc3cc(C)ccc3F)CC2)C1 C=CCCC(C(=O)NCC1CC12CCC2)NC(=O)CN1CCNC(=O)C1 CCC(C)CC(N)C(=O)Nc1noc(C(c2ccc(OC)c(OC)c2)C)n1 c1(OC)cnc(C(N2CC3(CC3)CC2CNC(=O)CCC2CC2(Cl)Cl)=O)c(F)c1 C1(NC(=O)Nc2nc(C(C)(C)C)c(C(F)(F)F)s2)CC2CCCCCC2C1 N1(C(C2(C)CC(=C)C2)=O)CCC(CO)(CNC(c2cccc(C#N)c2)=O)CC1 C(=O)(CCCCC(=O)OC)N1CCCC(O)(CN(C(=O)C(C)(C)N2CCCC2)C)C1 CN1CCC(CN(C(c2sccc2Br)C(=O)NCC2CCOC2)C)CC1 CCCC(C#N)C(=O)N1CC(NC(c2cc(OC)ns2)=O)C(n2cccn2)C1 CCC(C)(C)C(O)C(=O)N1CC(NC(c2cccc(C)c2N)=O)C(C)C1 Cc1cc(N)c(C(N2CCC(C)C2CNC(C2CSCC(=O)N2)=O)=O)c(F)c1 c1(C(=O)NCCCOCCN(C(=O)C=CSc2nc[nH]n2)C)cc(C2CC2)no1 c1(C(=O)NC(C)C(C)(C)C)coc2c1CN(C(=O)CC1(O)CCOCC1)C2 c1(SC)cccc(C(=O)NCC(C)(O)CNC(C2CCC(F)(F)C2)=O)c1[N+](=O)[O-] C1(CC=C)(NC(=O)CCC(C)OC)CCCN(c2nnc(O)s2)C1 c1(CN2C(C)C(c3ccccc3)CC2)ccnc(S(C)(=O)=O)c1 C1(NC(c2cn(CC(C)C)nc2)=O)CCCN(C(=O)Cc2csc(S)n2)C1C C12(NC(c3cc(C)on3)=O)CCCN(C(=O)C(=Cc3cccnc3)F)CC1C2 C(=O)(C(CCC)CC(C)C)NC(C(=O)N(CC#C)CCF)Cc1ccco1 CN1CCCC(N=c2ccnc(N3CCOC(c4ccccc4Cl)C3)[nH]2)C1 C(=O)(CCC(=O)N1CCCCC1C(=O)N(C)CC1CCCC2CC12)N(C)C C(=O)(CC(C(C)(C)C)NC(=O)C(C)OCCC(C)C)N1CC(CCC)C1 c1(CC(=O)NCCCC(C)NC(CCC(=O)NC)=O)coc2ccccc12 c1(C(C)=O)cccc(OC(C)C(=O)NCC(C)(C)NC(C2COC(=O)N2C)=O)c1 c1(OC)ccc2cnc(N3CCC(NC(c4cc(C)c[nH]4)=O)C(C)(C)C3)nc2c1 Cc1cc(C)c(CC(N2CCC3(NC(=O)C4=COCCC4)CC3C2)=O)c(C)c1 C(=O)(C(C)C(C)S(C)(=O)=O)NC1C2CN(c3ncnc(CC)c3F)CC21 c1(CC)cc(NC(=O)C2=CCC(NC(C3(C)CNC(=O)C3)=O)C2)cc(C)c1 C12(CNC(c3ccnc(O)c3Br)=O)CCCC1N(C(C1(O)CC1)=O)CCC2 c1(NCC2CCN(C(c3c(CC)nc(C)[nH]3)=O)CC2C)ncc(C#N)cc1C C=CCC(CC(C)C)C(=O)NCC1CC1C(N1CC(CO)CC1(C)C)=O C12(C(C)NC(=O)CN3CCCCCCCC3)CC3CC(CC(C3)C1)C2 C1(CC(=O)NCC(CNC(C2(COC)COC2)=O)O)Sc2ccccc2NC1=O N1(C(Cc2n(C(C)C)ncc2)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C=CI C(CCCN=[N+]=[N-])NC(COC1(C)CN(C(C2CCC(C(=O)OC)C2)=O)C1)=O C1(C(=O)Nc2cc(C(=O)C3C4(CC4)C(=O)N3)on2)(CC)CC2(CC2)C1.CCO.OC c1(C2C(C(N3CC(F)(F)CC3CO)=O)C2)ccc(Cl)c(Cl)c1 c1(CC(=O)NC2CN(C(C34CCCCC3C4)=O)CCC2F)ccc(Br)cc1F Cc1cc(C(N2CCC2CNC(=O)C2=CCCOCC2)=O)c(Cl)cc1N C(=O)(CC(C)c1cnn(C)c1)NCC1N(C(C(F)OC)=O)CC1 N1(C(C(C)c2cccs2)=O)CCC(C2CC2)(CNC(=O)C2=CCCCC2)C1 c1(C(=O)NCC(C)(O)CNC(=O)C=Cc2ccoc2)ccc2ncsc2c1 C(=O)(C#CC1CCCCO1)NC(CCNC(c1cn(CC)nc1)=O)(C)C CC1(NC(c2nocc2C2CC2)=O)CN(C(C2(C3CCCCO3)CCC2)=O)C1 c1(C(N2CCC(NC(C3C4COCC34)=O)CC2)=O)cc2cc(Cl)cc(Cl)c2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)C(=O)N1CC(NC(N)=O)C1)C N1(C(C2(C)CCNC2)=O)CCN(CC(N)=O)C(=O)C1.C(=O)(CCl)N N1(C(C(C)C2CCCOC2)C(=O)NCS(N)(=O)=O)CCC(S(=O)(=O)C(C)C)CC1 C1(CC(=O)NC(CNC(C(C)n2cccn2)=O)CC(C)C)CN2CCN1CC2 CC(C)CCC(=O)N1CC(C)CC1C(=O)NCC1CC(CN(C)C)C1 C1(NC(c2coc(Cl)n2)=O)CC(F)CN(C(=O)C=Cc2ccncn2)C1 c1(C(=O)NC2CC(C)(CNC(c3ccn(CCC)c3)=O)C2)nncnc1C C(=O)(C1=CS(=O)CCC1)N(CC(C)NC(=O)C=Cc1ccc(=N)[nH]c1)C c1(CC(C)C(=O)NC2CCCN(C(C3CC(C)(O)C3)=O)C2C)ccc(F)cc1F c1(N(C)CCOC2CC2)cc(N2CC3CCC3C2)nc(-c2ccncc2)n1 CCCC(CCC)CC(=O)N1CC(O)CC1CNC(c1cc2c(s1)CCCC2)=O C1(CC(=O)NCCC2N(C(CCCOCC=C)=O)CCC2)NC(=O)CNC1=O C1(C(N(C2CCOC2)C)=O)CCN1Cc1cncs1 CC(C)(CCS(C)(=O)=O)C(=O)N1CCC1c1cn(-c2ccccc2C(=O)O)nn1 C1(C(N2C(C3CCCN(C(=O)C=CCO)C3)CCC2)=O)Cc2nccnc2C1 N1(C(C2N(C(C(C)Cn3cccn3)=O)CC3CC32)=O)CCn2ncnc2C1 C(=O)(CCC(=O)NCC(C1CCC1)NC(=O)CS(N)(=O)=O)NCC c1(C(N(CC(CC)NC(C2CC3CC3C2)=O)C)=O)c(C)nn2c(C)cc(C)nc12 N1(C(c2cn(CCC=C)nn2)=O)CC2CN(C(=O)C(O)C(F)F)CCC12 Cc1cccc(Br)c1C(C(N1C2CCC1C(CO)C2)=O)NC(=O)C(C)O c1(C(=O)NC2C=CC(CC(=O)NC(C(C)(C)OC)C)C2)cc2cccnc2[nH]1 C#CCC(CC(F)F)C(=O)NC(CC(=O)NC1(C(C)C)CC1)C(F)F CC1(N(C(CCC2(C)CC2)=O)C2CCOC2)CCN(C(c2ccc(F)cc2)=O)C1 CN1CC2C(C(N3CC4CC3C4NC(=O)CCCCC3CC3)=O)C2C1 c1(C(N2CC(C)CC(OC)C2)=O)ccc2c(n1)CN(C(C1OCCC1C)=O)CC2 CC1CCN(C(=O)CSCc2ccnn2C)CC1NC(=O)C=CCN1CCCC1 N1(C(C2C(C(=C)C)OCC2)=O)CC2CC(C1)CN(C(=O)C(C)OC)C2 C(=O)(CCCC(C)(C)C#N)N(C)CC1C2CN(C(C3CN(CC)C(=O)C3)=O)CC21 C1(C(=O)NCCc2c(CNC(CC(C)OC)=O)nco2)CCCC1(C)C C1(CC(=O)NC(CNC(C2(CCC)CC2)=O)COC)COC(C)(C)C1 CC1CCCC1N(C(=O)C(C1(O)CN(C(c2cnc(O)o2)=O)C1)F)C O=C1C2=C(CCl)NC(=S)NC2c2cc3scc1c3s2.OC(F)F c1(C(=O)NCC2(O)CN(C(=O)CSCc3cccs3)C2)ccc2c(O)n[nH]c2c1 c1(CNC2CC(C(N3CCn4ncnc4C3)=O)C2)c(Cl)cc(Cl)nc1Cl CC(O)(C(=O)N1CCCC1C1CCN(C(c2ccc(F)c(F)c2)=O)C1)C(F)(F)F c1(C(CCC)C)nc(-c2oc(C(F)F)cc2C)n(CCOCC)n1 C(=O)(C(C)CC(=O)NCC1CCN(C(=O)CCNS(C)(=O)=O)C1)OC c1(NC(CC=C)CC(C)C)c(Cl)ccc2c(C)cc(=O)oc12 C(C)(C(C(=O)OC1CC1(c1ccccc1)F)N(C)C)OC C(=O)(CCC(=O)N1CCC(O)CC1)N(CC(C)N(C(=O)CC1CCCCC1)C)C c1(C(=O)NC2(CNC(C3CC(=C)C3)=O)CCCCC2)ccc2c(c1)CCC2(C)C c1(N(C)CC2CCN(C(C3(O)CC(C)(C)C3)=O)C2)nc2ccccc2o1 c1(C(=O)OC)ccc(C(=O)NC(C)CC2CN(C(=O)CC3CCCC34CC4)C2)cn1 CC1CCN2N=C(C(=O)NC3CC3NC(C3CC3c3ccc(Cl)cc3)=O)NC2=N1 C1(C(=O)NCC=CCNC(C2(O)COC2)=O)C2CCC1(c1cncs1)C2 N1(C(Cc2cn(C(C)C)nc2)=O)CC(NC(=O)CCc2ccn(C)n2)C2(CC2)C1 c1(C(N(CCC(C)NC(c2cnc(C)[nH]2)=O)C)=O)nnccc1C(F)(F)F c1(C(N2C(C)CCC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)cnn2ncccc12 c1(COC)cncc(C(N2CCCCC2C(C)(C)NC(c2csc(Cl)n2)=O)=O)c1 Cc1cccc(Br)c1C(C(=O)Nc1ccc(Cl)cc1)NC(=O)CC1CC2(CC2)C1 C1(CC)CCCC1(C)C(=O)NCCC1(CNC(c2ccnn2C(C)(C)C)=O)CC1 CCCCC(C)N(C(=O)C=CC1(C)CN1)C.C(CCCC)N CC1(O)CCN(C(C2C3CCN(C(=O)CNC(C4CC4C)=O)CC23)=O)CC1 N1(C(C2CC(SC)C2)=O)CCC2(CCCN2C(c2cccnc2OC)=O)C1 C1(CC)(NC(c2ccc(OC)nc2C)=O)CCN(C(=O)C(O)C(F)(F)F)CC1 C1(C(N2CC(C)N(C(=O)CC3CN(C)C3)CCC2)=O)CCc2ncccc2C1 N1(C(CC)C)CCC(n2cc(C)cn2)CC1.N12CCC(CC1)C2 C1(C(N2CC(CCCCNC(C3ON=C(CC)C3)=O)C2)=O)CC2(CO1)CC(F)(F)C2 c1(CNC(C2CC(=O)N(C3CC3)C2)=O)cnn2c1CN(CC(O)CC(F)(F)F)CC2 C1(C(=O)NC(C)(C)CNC(c2ccc(Br)cc2N)=O)CCc2cncn2C1 S(=O)(=O)(c1cccc(Cl)c1)N1CCCC(F)(CNC(C(C(C)C)O)=O)C1 CC1CCCN(C(c2cc(CNC(c3cnc(O)o3)=O)[nH]n2)=O)C1 C1(CNC(CNC(CNC(C2(COC)CCCO2)=O)=O)=O)CCC=CCCC1 Cn1nc(C(N2CCC(CNC(c3nc(C4CC4)cs3)=O)C2)=O)c(C(F)F)c1Cl C(C(O)C(=O)NOC1CC2CCC1C2)=CC.n12cc(nn1)COCC2 C1(NC(CC(C)OC)=O)CC2CCCC(C1)N2C(c1[nH]nc([N+](=O)[O-])c1Cl)=O N1(C(C2(CC)CCCO2)=O)CC2CCC1CN2C(C1OC2CCCCC2C1C)=O C1(NC(C2NCC(N=[N+]=[N-])C2)=O)CCC2(CC1)C(C(=O)O)C2(F)F c1(OCc2cn(C(CC=C)CC)nn2)c(C)cc(C)cc1C c1(C(N(C)CC2CCN(C(C3CNC(=O)C3)=O)CC2)=O)n[nH]c2c1CCC2 c1(OC)nc(C)ncc1C(=O)NCC1(F)CCN(C(=O)C=CSC)CC1 N1(C(CNC(=O)NC)=O)CCN(C(C2CCOC(C)C2)=O)CC1.C12(C)CC(C1)N2 C1(C(N2CCN(C)C2=O)=O)CC12CCN(C(C1CC(OC3CC3)C1)=O)C2 C1(C(=O)NC2CCC(NC(c3c(C)ccnn3)=O)CC2)CCN2CCC1C2 N1(C(c2cnc(C#N)s2)=O)CCCC2(CCCN2C(c2ccncn2)=O)C1 N1(C(C(C)OCCC#C)=O)CC2(CCCN(C(C3CCCCN3CC)=O)C2)C1 c1(C(C)C)cc(C(N2CCC(CNC(c3c[nH]c(Br)c3)=O)C23CC3)=O)cc(O)n1 C1(C(N2CCC(NC(c3cncc(OCC)c3)=O)(CF)C2)=O)CCOC(=O)CC1 C(C(C(=O)NOCCCC(F)(F)F)OC)NC(C1CC(CC)C1)=O Cc1cc(C)c(C=CC(N2CC(NC(C3(O)CC3(C)C)=O)CC(F)C2)=O)cc1C c1(-n2cc(CSCCNC(C3CC4C=CC3CC4)=O)nn2)cc(Cl)c(F)cc1F C(=O)(C1=COCCC1)NC1CC(NC(=O)CC2CCC3CC3C2)C1 C1(C(=O)N(C)CC2COCCO2)(NC(c2n(CC)nnc2)=O)CCCC1C C1(NC(=O)NC2C(SC)COC2)CC12CCc1cc(Br)ccc12 c1(OC)c[nH]c(C(=O)NC2CCN(C(c3ccc(C)s3)=O)C(C)C2)cc1=O CCC(C)CCC(=O)NC1(C)CCN(C(c2cc(OC)ccc2C(C)C)=O)CC1 CCCC(C)CC(=O)NCCC1CN(C(c2c(C)noc2C2CC2)=O)CCO1 C(=O)(C(C#N)C(C)C)N(CCNC(c1cnc(C(C)O)s1)=O)CC C(=O)(C1c2c[nH]nc2CN1C(=O)C(C)N(C)C1CC1)NS(CCC)(=O)=O N1(C(C2(C=C)CCC2)=O)CCCOC(CNC(C2CCC(C)(C)CO2)=O)C1 c1(C(C(=O)NC)N(C(c2cccc(Cl)c2)CCO)C)cc(C)cc(C)c1 C(=O)(C1=CCC(C)CC1)NC1CC(N(C(c2cc(C)c(Br)s2)=O)C)C1 c1(C(=O)NC(CCOC)CNC(c2nc(C)ccc2C)=O)snc2ccccc12 CC(CF)N=c1ccc(Br)c(S(=O)(=O)N2CCC(Oc3ccncc3)C2)[nH]1 N1(C(=O)NCc2nc3c(Br)csc3s2)c2ccncc2N2CCC1C2 CC(CC(=O)N1CCCC1CNC(=O)CCc1nnc(C2CC2)o1)CC(C)(C)C c1(C(=O)NC(C2CCN(C(c3nc(CC)oc3)=O)CC2)C)ccc(S(C)=O)cc1 c1(C(=O)NCCC2(C)CCN(C(CCN(C)CC)=O)C2)c(Cl)ccc(C)c1N c1(C(c2nn[nH]n2)=O)cc(-c2ccccc2SC)c(NC2C(CC)C2)cc1OC CC1CCN(C(C2CC=CCC2)=O)CCN1C(=O)CNC(=O)CC1CCCCC1 c1(C(N2C(CN(C(=O)CC3CSCCS3)C)CCC2)=O)ccc(F)s1 C1(CNC(=O)CNC(c2cccs2)=O)C=CC(NC(=O)COCCO)C1 Cc1nn(CC(=O)NC(C)CC2CN(C(=O)CC3COCCO3)C2)c(=O)n1C Cc1cnc(F)c(C(=O)N(C(C)CNC(c2nn(C)cc2N)=O)C)c1 N1(C(C(COC)COC)=O)CCC(CO)C(NC(=O)CCN2CCNC(=O)C2)C1 c1(C(N2C(CCNC(c3c(Cl)cc(C)s3)=O)CSCC2)=O)cnn2ccsc12 C1(C(=O)NCC#C)CCC2CCC1N2C(=O)CN1CC(=O)NC1=O N1(C(Cc2c(C)noc2Cl)=O)CC(NC(=O)C(C2CC2)N(C)C)C(C)(C)C1 C(=O)(C1=CCCOC1)N(C(C)CCNC(c1ccnc(SC2CCC2)c1)=O)C CC(CC(F)(F)F)C(=O)NC1CCCN(C(=O)COC(=O)N(C)C)CC1 N1(C(=O)NCc2ccccc2N2CCOCC2)CCC(C2CC2(F)F)C1 C=CCC(CC)C(=O)N(C(C)(C(=O)NCc1ccsc1)C1CC1)C C1(NC(=O)Nc2c(C)ncc(C(=O)NC)c2)CC(C(C)=NO)C1(C)C CC1CC(C(=O)N2C3CCC2(CNC(C2Cc4nnsc4S2)=O)CC3)=NO1 N1(C(C)=O)CC2CN(C(=O)Cn3cc(C)cn3)CCC12.C(=O)CCC C1(C(NOCC(=O)NCC2CCC(C)(CC)O2)=O)CCC(C2CC2)C1 Cc1c(C(N2CCCC(N3CCN(c4ncncc4Cl)CC3)C2)=O)cccc1Cl c1(-c2ccc(CC)c(F)c2)c[nH]c2ccc(C(=O)Nc3cc(O)ncn3)cc12 C1(NC(C2(O)C(C)(C)C2)=O)CN(C(c2ccc(F)c(F)c2N)=O)C2(CCC2)C1 N1(C(C2CC(C)(F)C2)=O)CCC(CO)C(NC(=O)C=Cc2cscn2)C1 C(CC(C)(C)CC)(C(=O)NCC)N(CC#C)C.C1C(=O)N1 N1(C(c2cc(SC)oc2)=O)CCOC(C(=O)N(C)Cc2nncn2C)CC1 c1(OC)cc(C(=O)NCC2COCC2NC(=O)COC(C)(C)C)[nH]n1 C(=O)(C(CCN(C)C)NC(c1cc(C2CC2)[nH]n1)=O)N1CC(C(C)O)C1 c1(C(=O)NC2(C)CN(C(c3c(C)ccc(OC)n3)=O)C2)cccc2ccnn12 C=Cc1ccc(CNC2CN(C(C3CCC(CC)CC3)=O)CCC2F)cc1 CCC(C)(CO)C(=O)N1CCC(OC2CN(C(C3CN(C)C(=O)N3)=O)C2)CC1 Cc1cnc(C2CN(C(C34CC(CN3C(=O)CCCF)C4)=O)C2)nc1 c1(N2CCN(C)C(CNC(C3CCCNS3(=O)=O)=O)C2)nc2cccc(F)c2o1 c1(C(C)NC(=O)Cc2cccs2)ccc(CNC(c2ncn(C)n2)=O)cc1 c1(C(=O)NCC(C)(C2CC2)NC(C2C(C)=C2)=O)cnc(Cl)c(C2CC2)c1 N1(C(C2CC(C)OC2)=O)CCC(Nc2ccncn2)CC1C CC(CNC(=O)OC(C)(C)C)CC(=O)N1CCC(N(C(=O)Cc2cn[nH]c2)C)C1 C1(NC(COCCCCCC)=O)CC2(CCC2)CN1C(=O)CCCc1cccs1 N1(C(C(C)CF)=O)CC2CC2(CNC(c2cn(C)nc2-c2cccnc2)=O)C1 c1(SCC(=O)NC(CC=C)CNC(=O)C(C)c2cc[nH]n2)cccc(OC)c1 c1(C(=O)NC2(C)CCCN(C(Cc3cc(C)no3)=O)C2)nn2ccccc2c1C c1(NC(C2(C)CCCOC2)=O)ccc2c(c1)CCCNC2 C(CC(C(=O)NCCCN1CCCC1)NC(=O)CNS(=O)(=O)CC)=CC CC(C)CC(C(=O)N(C1CC2CC2C1)C)ONC(C1C(C#N)C1(C)C)=O CC(C)C(CNC(c1cnn(CCF)c1)=O)NC(C1(C(F)F)CCCC1)=O c1(N2CCC(N(C(C(C)=C3CC3)=O)C)CC2)nc(C)nc2sc3c(c12)CCCC3 N1(C(C)=O)CCC(C)(C(=O)NC2(CO)CCCCC2)C1.c12ccc(s1)c(=O)[nH]2 C#CC1(C)CCCN(C(=O)C(Cn2cncn2)NC(c2cnn(C)c2Cl)=O)C1 C1(C)(OCC(=O)OC)CNC(=O)C2CCC(CC2)NC1=O.C1(N(C)C)CCCC1 c1(C(=O)NC(CNC(c2nccc(CC)c2)=O)C(C)(C)C)cc(C)n(C)c(=O)c1 Cc1cncc(C(=O)NC23CC(NC(c4ccc(OC5CCCC5)cc4)=O)(C2)C3)c1 c1(C(=O)NC(CC)C)ccc(C2CCCN(CC3CC3(C)C)C2)cc1 C(=O)(C1CCCc2nccn21)NCC(CNC(C(C)(C)CF)=O)CO Cc1cc(C#N)ccc1C(N1CCC(C)(CNC(=O)C=CI)C1)=O C1(C(N2CC(CNC(C(CCOC)C)=O)OCC2)=O)CN2CCN1C(C)C2 C(c1cccc(Cl)c1)=CC(N1CCC(NC(C(CCC)=CCC)=O)(COC)C1)=O C1(CNC(c2nnc(C(C)C)s2)=O)COCCN1C(=O)C(C)c1cc[nH]n1 c1(CC)ncc(C(=O)NCC2(CO)CCN(C(=O)C(C)(O)COC)C2)c(C)n1 C(N=c1cc(Br)n(C)[nH]1)(c1nnnn1C1CCOC1)Cc1scc(CCC)n1.SC CC1CN(C(=O)Cc2cnnn2C)CC(CCNC(=O)CN2CCCC2=O)O1 Cc1nc(=N)[nH]cc1C(=O)NC(C1CCN(C(C2CC(=O)N(C(C)C)C2)=O)C1)C c1(C2(N3CCCC(C(N4C(C(=O)OC)C(C)C4)=O)C3)CC2)cn2ccccc2n1 N1(C(C(C(C)C)CO)=O)CC(NC(=O)C(C)OCC2CC2)CC2(CCC2)C1 CCC(c1ccc(OC)cc1)=CC(=O)N(C)CC1CCCN1C(=O)CCCOC c1(CC)nc(C)n(C)c1C(=O)NCC12CC1CN(C(C1NC(=O)OC1C)=O)C2 C(=O)(C1=NOC2COCC12)C(=O)Cc1ccsc1.C1(C(CN)N)CCCC1 c1(-c2nc(CC)on2)cccc(CNCC2CCCN2C(c2cc(Cl)c[nH]2)=O)c1 c1(C(=O)N(c2ccccc2)CCO)csc2cccc(-c3nn[nH]n3)c12 C1(S(N)(=O)=O)(C(=O)NCCCC2N(C(CCS(=O)(=O)NC)=O)CCC2)CCCC1 c1(C(N2CC(NC(C(C)CN(C)C)=O)C3(C2)CC3)=O)c(N)cc(Cl)cc1Cl N1(C(CN(CCC)C)=O)CCC(O)(CN(C(=O)Cc2cc[nH]n2)C)CC1 C1(O)(CNC(c2cc(SC)nn2C)=O)CCCN(C(=O)C(C2CCOCC2)F)C1 Cc1cc(C(=O)NC23COC(CNC(=O)C(O)CN(C)C)(C2)C3)cc(C)n1 c1(CC)cc(C(=O)NCC2CCN2C(=O)Cn2nnc(SC3CC3)n2)c(C)o1 C(C(C(C)C)C(C)C)NNC.c12ccc(c(F)c1)C(C(=O)NC1CC1)N2C c1(C(=O)NC(C)CC(C)NC(=O)C=Cc2cccc(F)c2)ccc(P(C)(C)=O)o1 C(=O)(CCS(C)(=O)=O)NCCCC(C)NC(C12CC(CF)(CO1)C2)=O C1(N(C(C2(CCOC)CC2)=O)C)CCN(C(=O)C=CCN2CCCC2)CC1C CC(C)CCCCCC(=O)N1CCC(F)(F)C(CNC(=O)C(F)(F)C(C)O)C1 S(=O)(=O)(c1c(Br)nc(C)n1C)N1C(Nc2cccc(C)c2)CCC1 CN1CCC2CCN(C(C3CC4CN(C(=O)CC5CC(F)(F)C5)CC4C3)=O)C2C1 c1(C(N2CCC(CCNC(C3CCC3(F)F)=O)C2)=O)cccc(C2(F)COC2)c1 c1(C(=O)NCC2CCN(C(C3N(C(N)=O)CCC3)=O)CC2)cc2cc[nH]c2cn1 C(=O)(C1=CC2(CCOCC2)C1)NCC1CN(C(CCN(CC)CC)=O)CC(C)O1 N1(C(c2n(CCN(C)C)ncc2)=O)CCC(NC(=O)CCS(C)=O)C(CO)CC1 C1(C(=O)NC2CN(C(c3csc(C)n3)CC)C2)(C(=O)OC)CCOCC1 N1(CC(C)C)N=C(C(=O)NC2CCCC(NC(=O)CO)C2)CCC1=O c1(C(=O)NCC(CNC(c2c(C)scn2)=O)O)cc2c(C)cccn2c1 Cc1nc(CC(=O)NCCNC(C2CCC(C(=O)OC(C)(C)C)C2)=O)c(Cl)s1 c1(C(=O)OCC(=O)Nc2c(OC)cccc2)cc2n(c(=O)c1)CCS2 C12(NC(=O)C=CC3CCOC3)CCC(CC1)N(C(c1cc(F)c(F)c(F)c1)=O)C2 C1(CNC(C(C)=C2CCCC2)=O)CC2CC(C1)N(C(=O)C=Cc1sccc1C)C2 Cc1ccc(C(=O)NCC2(O)CC(NC(=O)C(C)n3ccnc3)C2)c(Cl)c1 C1(NC(Cn2nnc(C)n2)=O)CC2CCC1CC2NC(C1CCCC(=O)O1)=O Cc1c(Br)noc1C(=O)NCC1CCN1C(C1CC1(F)F)=O CCC(C)C(O)C(=O)NC1(CNC(c2ccc(C(N)=O)c(Cl)c2)=O)CC1 Cc1cnc(CC(=O)NCCC(C)NC(c2c[nH]cc2C2CC2)=O)s1 C1(C(N(C)CC2CC(=C)C2)=O)C=CCN1C(C1CCS1(=O)=O)=O c1(C=O)ccc(N)c(F)n1.N1(CCC(C)C(=O)NCCNC(=O)C2CC2)CCC(C)C1 C1(NC(CCOC(C)=O)=O)CCN(C(c2cccc(C)c2C)=O)CC1O c1(CC2(C(=O)NC(CNC(=O)CC3CCCOC3)C3CC3)CC2)cccc(Cl)c1 C1(CCNC(C2(Sc3ccccc3)CC2)=O)(CNC(C2(O)CC2)=O)CCCC1 C1(C(N2C(C(C)C)CN(C(=O)C(O)CN(C)C)CC2)=O)OCCOC12CCC2 c1(C(N2CCC(NC(C3CN(CC(F)(F)F)C3)=O)C2)=O)cn2ccnc2s1 c1(C(C(C2=CCSC2)c2nnnn2N)C)ccc(F)cc1.c1(SCO)nnn(C)n1 C=C(C)CCN=c1nc(N2CCC(OCCF)C2)c2c(ncn2CC)[nH]1 Cc1cc(C(=O)NCC(C)N(C)C(c2cc(C3CC3)[nH]n2)=O)cc(Br)c1 Cn1c(CCNC(=O)C(C)(C)c2ccc(Br)s2)nc2cc(Cl)ccc12 c1(C(=O)NCC(C)(O)C(=O)O)c[nH]c2c(F)cc(F)cc2c1=O n1(CC(=O)NCC2(OC)CN(C(=O)C(C)CSC(F)(F)F)C2)cnc([N+](=O)[O-])c1 c1(C(=O)NC(c2nc(C(=O)N(C)CCn3cccn3)co2)C)ncccn1 Cc1cc(C(C)(C)C)c(C)cc1NC1(c2nnnn2C2(C)CC2)COCCC1C C1(C(=O)NC2CN(C(C(=C(C)C(C)(C)C)CC)=O)CC(O)C2)CN2CCCCC2CO1 Cc1csc(C(N2CCCC2CN(C)C(C2CC2c2ccnn2C)=O)=O)c1 c12cc(C(=O)NC)cc(n1)NC2=O.C1(CC=C)(C(=O)OC)CC1 Cn1nc(COc2ccccc2Cc2ccccc2)c(I)c1C(F)(F)F c1(SCC(=O)NCC2(OCC)CCC2)cn(CC2CCCOC2)nn1 C1(CCNC(c2n[nH]cc2Br)=O)(NC(c2ccsn2)=O)CCCC1 N1(C(C(C(C)C)c2ccncc2)=O)CCC(C)N(C(C2CC(C)(C)CO2)=O)CC1 N1(C(c2ncc(OC)nc2)=O)CCC(NC(C2(n3cnnn3)CC2)=O)C(O)C1 N1(C(C2C(CNC(C(C)OCC#C)=O)CCCC2)=O)CC2CC3CC2C1C3 c1(C(N2C(CCNC(=O)CC3(CO)CC3)CC(F)(F)C2)=O)ccc2ncnn2c1 CC1(C(=O)NC(CCO)C(F)(F)F)CC(O)CN1C(c1ccc(F)c(F)c1)=O CC(C)(C(=O)N1C2CCC1CC(NC(C1(F)CCCC1)=O)C2)C1=CCSCC1 C1(CNC(=O)Cc2cscn2)CN(C(C2(C(F)F)CCC2)=O)CCC1C(F)(F)F c1(C(N2CC3CN(Cc4cccc(I)c4F)C3C2)=O)c(F)cc(F)cc1Cl C1(C(C)NC(c2c(C)nc[nH]2)=O)CN(C(C2CC2CN(C)C)=O)CCO1 CC1CN(C(=O)C=C2CCSCC2)CC(C)C1NC(=O)CC12CCC(CC1)C2 C#Cc1cnn(C)c1C(=O)NC(C(=O)NCC(N)=O)C(C)CC c1(OC)cc(CNc2cc(N(C)CCC3CCCCC3)ncn2)ncn1 C1(NC(=O)CCn2cncn2)CC2CCN(C(=O)N=c3cccn[nH]3)CC12 CCC(F)(F)CC(=O)N(CCCN(C(=O)CCc1cc(OC)no1)C)C N1(C(C)=O)CCCN(C(=O)C(C)COC)CC1.C12(C(=O)NC)CSCC1C2 Cc1sc2ncc(C(=O)NCCCC(C)(C)NC(=O)C(O)C(F)(F)F)n2c1C c1(C(C)C(=O)NC(C)(C)CNC(C2CC=CCO2)=O)ccc(Br)cc1 C(CCC(C(=O)NC(c1cnccn1)C)NC(C1CC=CC1)=O)OC Cc1cc(NC(=O)CC2COCCN2Cc2cccc(Cl)n2)c([N+](=O)[O-])cc1Br N1(C(c2cnc(=N)[nH]c2)=O)CC2CC(NC(C3CC4CCC(C3)S4)=O)C2C1 O=[N+]([O-])C1CCC2(CC1)CC2Nc1ccnc(N2CCc3cccc(N)c3C2)n1 C1(C(N(CCCc2nc(C)on2)C)=O)C2CN(C(C3CC4CC4C3)=O)CC12 O=S(=O)(CCCN1CCC(F)(c2ccccc2Cl)C1)c1ccccc1 C1(c2ccccc2)(C(=O)OCCC(C(=O)NC)NC(=O)NCC)CC(CC)=NO1 C1(CCNC(C2(C(=O)OC)CC(=C)C2)=O)C2CCC(C2)N1C(=O)CCC(CC)OC c1(C(=O)NCC2(NC(c3ccc[nH]3)=O)C(C)CCCC2)ccn2cncc2c1 C1(SCC(C2CCCCC2)C2CCCC2)CCCN(OC(C(C)(C)C)=O)C1 c1(C(=O)NC(C(C)(C)C)C(F)(F)F)cc([N+](=O)[O-])ccc1-n1cnnn1 c1(OC(C)C(=O)NCCN(C)C(c2ccc(CO)s2)=O)ccc(Cl)c(Cl)c1 N1(C(C(C(CC)O)(C)C)=O)CC2(CCCN(C(c3cc(C(N)=O)c[nH]3)=O)C2)C1 c1(OC)cccc(C)c1C(N1CCC(C(=O)Nc2ncc(C)c(Cl)n2)C1)=O N1(C(CC(C)(C)NC(C2CC2C2(C)COC2)=O)=O)CCC2(CNC(=O)O2)C1 Cn1cc(CNC(C2CC2C(F)F)=O)c(CNC(=O)C(C)(C)N2CCCC2)n1 C1(NC(C=CS(CC)(=O)=O)=O)CCC2CN(c3nc(C(C)C)nc(=N)[nH]3)CC2C1 c12ncnc(c1C)CNC(=O)C(C1(OC)CCC1)N2.C1(OC)CC(NC(C)C)C1 c1(OC)ccc(OCC(N2CCN(C(C3C=CCC3)=O)CC2C)=O)c(C)c1 C1(C(=O)NC(CN(C(c2cc(SC)oc2C)=O)CC)C)CC2CCC(C1)O2 c1(CC(=O)OC)ccc(-c2ccc(C3CC(=O)N(C)C3=O)cc2)c(C)n1 N1(C(C(C)(C)NC(=O)OC)=O)CCCCC1CCNC(=O)C(C)(C)c1ccsc1 CCCC(CCCNC(=O)CCc1ccc(N)cn1)NC(=O)C=Cc1ccc(Cl)s1 c1(C(N2CC(NC(c3c(C)n[nH]c3)=O)C3(C2)CCC3)=O)cc([N+](=O)[O-])ccc1C CC(C)CC(C)CC(=O)N1CCC(C(C)(C)NC(c2cncc(F)c2)=O)CC1 c1(C(N(CCC)CCNC(=O)C(O)C(C)OC)=O)c([N+](=O)[O-])ccc(C)c1C c1(OC(c2ccc(OC)c(Cl)c2)=O)cc(F)ccc1S(C)(=O)=O C1(CNC(C2C(C=C)C2)=O)CN(C(c2ccc(C3(C)CC3)cc2)=O)CC12CCC2 C(=O)(C(CCC(N)=O)n1cc(CO)nn1)N(C1CCN(C(=O)C2=CCSC2)CC1)C C1(C#N)(C(=O)NCC2N(C(Cn3nnc(C)n3)=O)CC(O)C2)CC12CCOCC2 c1(SCC(=O)NCC2C(NC(C3CCC(C)(C)O3)=O)CC2)ncnc2[nH]cnc12 N1(C(CC2(CSC)CC2)=O)CCCC2(CCCN2C(=O)CCc2nccn2C)C1 N1(C(c2n(CC)ccn2)=O)CCC2CN(C(=O)CCOC)CC12 Cn1[nH]c(=NC(=O)NCC2CCC(O)(C(F)(F)F)C2)cc1C#N C(=O)(C(C)C(C)(F)F)N1CC(C(C)NC(c2ncc(N(C)C)cn2)=O)C1 CC1(C)OC2(C(N3CCCCCC3CNC(=O)Cc3ccccc3)=O)CC1C2 Cc1cccc(CC(=O)NCCOCC(=O)N(C2CC2)CC2CCC(C)O2)c1 C(=O)(C(F)CC(C)(C)NC(c1cccnc1O)=O)NCc1cc(C)ncc1 c1(OC)ccc(C(C)N(C2CCCCC2)C(c2ccc(Br)cc2OC)C)c(C)c1 C1(C(=O)NC(Cn2cccn2)C(=O)NCCC2(CO)CCCC2)(CC)CCCC1 Cc1cc(Cl)nc(Cl)c1C(N1CCCC(C(=O)NC2CCC(=O)NC2)C1)=O N1(c2nc(Nc3c(CC)ccc(Br)c3)nc(C)c2)CCN2CCCC2C1 C1(C(=O)Nc2c(OC)cc(Br)c(C)n2)CCC(N=c2ncnc3[nH][nH]c(I)c2-3)C1 N#Cc1cc(C(N2CCCC2CNC(=O)Cc2ccc(Cl)cc2)=O)co1 C1(N(C(C(C)NC(N)=O)=O)C)CN(C(=O)Cc2ccn(C3CCCC3)n2)CC1F C(=O)(C1Cc2ccc(Cl)cc21)NCC(C)(CO)NC(c1cn(CC2CC2)nn1)=O c1(-c2ncc(C(=O)NCC3CN(c4ncc(F)cn4)CCO3)s2)cccnc1Cl c1(C(=O)NC(C2CN(C(c3cnsc3)=O)CCO2)C)ccc2c(c1)CC2 C1(CC(=O)N(C(CC)CO)C)C(NC(c2c[nH]nc2C)=O)CC1O CC1CCC(C)N1C(C)C(=O)NC1COCC1NC(c1ccccn1)=O c1(C(N2CC(NC(=O)C(C)(O)C3CC3)CC(OC)C2)=O)coc2c1C(=O)CCC2 N1(C(c2nc(C)sc2)=O)CC2(CCC2NC(c2cnc3sccn23)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CC2N(C(=O)NCc3c(CC)onc3)C(CC2)C1 C1(NC(CC(C)C)=O)(CNC(c2n[nH]cc2C(C)C)=O)CC2CCC1CC2 C1(NC(C2C(C)C2C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)CC(C)(C)C1 C(C(CC)CC)N(C(=O)C=C(C)CNC(=O)C(C)CC1CCC1)CCC S(=O)(=O)(c1cc(Br)cc(Br)c1)NCC1CCC2(CN(S(=O)(=O)CCBr)C2)CC1 N1(C(c2cccnc2Br)C(=O)NC2CC3C=CC2C3)CC=C(CCCO)CC1 c1(C(N2CCC(n3cc(CNC(c4cnccn4)=O)nn3)C2)=O)cc(Cl)c(Cl)s1 CCC(CN(C)C)CC(=O)NC1CC(F)(CNC(=O)CSC2CCCCO2)C1 N1(C(C2=NOC(CNC(c3cncc(OC)c3)=O)C2)=O)CCC2=C(CCCC2)C1 N1(C(C2(CC(C)C)CCC2)=O)CCOC2(C1)CN(C(=O)CC1CCCC(C)C1)C2 S(=O)(=O)(c1cc(C(=O)NCC(C)(C2CC2)NC(=O)CCC2CCCO2)co1)NC c1(C(N(CC(CN(C(=O)Cc2nncn2C)C)O)C)=O)cccnn1 CCC(CC(=O)NCC1CCCCC1NC(c1ccc2ccnn2c1)=O)C(C)C C(=O)(CC(C)n1cc(Br)cn1)NCC1CC(NC(CSCCOC)=O)C1 C1(C(N2CCN(C(C(CCC)OC)=O)CC2)=O)CCCN(S(N)(=O)=O)C1 N1(C(C(C2CCC2)OC)=O)CCC(CNC(=O)C(=O)N=S(C)(C)=O)C(F)(F)CC1 Cc1nocc1C(=O)NC(C1CCN(C(C2CCC(N(C)C)C2)=O)C1)(C)C c1(C(N2CC(OCC)(CNC(=O)C(C)CO)C2)=O)cnc2c(c1)CCS(=O)(=O)C2 C1(NC(C2N(C(C)C)C(=O)CC2)=O)CCN(C(=O)CC(C)C2CC2)C12CCCC2 CCC(C)CCCC(=O)NCCCN(C(=O)Cc1c(C)nn(C)c1C)CC1CC1 C1(C(C)C(=O)NCC(C)N(C)C)CCN(C(C2CCC2C#N)=O)CC1 C1(OC)CC(CNC(=O)C(O)Cc2ccccc2)N(C(=O)Cn2ccc(C)n2)C1 c1(C(N(CC(C)NC(=O)C(c2cnccn2)C)C)=O)ccc(OC(F)F)cc1F N1(C(C(C)=CCC)=O)CCC(C(=O)Nc2cccc(F)c2CC)C(C)C1 C1(NC(c2c(C)cn(C)c2)=O)CC(O)CN(C(c2ccc(C(C)O)cc2)=O)C1 Cc1nc2[nH][nH]cc-2c(=Nc2ccc(CC(=O)NCCF)cc2O)n1 C(=O)(C1CC=Cc2ccccc21)NCCC(C)NC(=O)COC1(C)CCOCC1 Cc1n[nH]c(C)c1C(C)CC(=O)NCCCC1CCCN1C(=O)C1=CCCO1 N1(C(c2c(OC)cc(F)cc2)=O)C(C)CC2CN(C(=O)CCCCC(C)C)CC12 C1(C(=O)NCCCn2cc(-c3cn(C(C)C)nc3)nn2)CCCC12CC2 C(=O)(C(C)S(C)(=O)=O)N1CC(C)C(CNC(C2COC(=O)O2)=O)C1 N1(C(COCCC#C)=O)CCC2(C(=O)NCC3OCCCC3(C)C)CCCC12 c1(OC)ccc(C(=O)NC(C2(O)CCN(C(=O)CCSC3CC3)C2)C)c(OC)n1 c1(NCC(=O)NC2C(CNC(c3cc(SC)oc3C)=O)C2)ccc(C#N)cc1 c1(COC)cc(C(=O)NC(C)C(=O)NCCN2CCOCC2)n[nH]1 FC(F)(F)CCN=c1nc(N2CCC(c3cccnc3)C2)c2cccc(F)c2[nH]1 C1(NC(C(C(=C)C)(C)C)=O)COC2(CCCN(C(=O)CCn3cncn3)C2)C1 C1(C(N2CCCN(C(C(C)CO)=O)CCC2)=O)Cc2cccc(OC(F)F)c2O1 C1(CNC(c2c(C)ncnc2)=O)CCCC2(CN(C(=O)Cc3c[nH]nc3O)C2)O1 n1(CCC(=O)NC2C(CNC(=O)C3=CCCS3)C2)c(=O)nc(O)c2ccccc12 C1(NC(C(COC)C)=O)CCCN(C(=O)Cc2c(Br)cnn2C)C1 c1(CC(C(=O)NCCOC)NC(C2CCC(=O)O2)=O)ccccc1Br N1(C(CN(c2ccccc2)CCC#C)=O)CC(O)CCC1c1ccccc1 C1(C(=O)NCCC2(O)CN(C(COCCC#C)=O)C2)(OC)CCC12CCC2 CC1CN(c2cc(N(C)Cc3nnc(O)o3)ncn2)Cc2nncn21 Cc1ccncc1C(=O)NCC12CC1CN(C(=O)C(N1CCCC1)C1CC1)C2 Cc1nn(CC(=O)O)c(C)c1CN(CCNCC1(F)CCOC1)C N1(C(C(C)N(CC)CC)=O)CC(CO)C2(C1)CN(C(C1CC3(CSC3)C1)=O)C2 N1(C(C2CC(C)(C)C2)=O)CCC2CCN(C(c3cc(F)c(O)c(Cl)c3)=O)C2C1 c1(CC)ncnc(N2CCCC(CC(=O)Nc3ccc(OC)c(Br)c3)C2)c1F c1(NC(C2C(NC(C=Cc3ccc(C)s3)=O)C2)=O)ccc2c(c1)CCCC2=O c1(C(=O)NCC(CNC(C(C)OCOC)=O)O)cccc(C)c1Br C1(CC(=O)NC2CCC(NC(c3c(C)nc(C(C)C)o3)=O)C2)COC(C)(C)CO1 C#CCC(C)(C(=O)NCC(C)CSC)NC(=O)C(=O)N(C)C c1(NC(=O)NC(CC#C)COC)cc(-c2ccccc2)nn1-c1ccccc1 N1(C(CCCCCOC)=O)CCCC2(CCN(c3ccc(OC(C)C)cn3)C2)C1 Cc1ncc(C(=O)N(C)CC2CCCN2C(=O)CNC(=O)NC(C)C)n1C(F)F N1(CC)C(=O)CCC1C(N1CCC(NC(c2cn(CC)cn2)=O)C1)=O CCCC(CC(C)C)C(=O)NC(C(N1CCCC(NC(N)=O)C1)=O)C1CC1 N(C(=NCC1(C#N)CCOC1)NC1C2(CC2)C12CC2)C(C)C c1(NC(COCCOCC#C)=O)ccc(N)c(CNC(C2(C(C)C)CCC2)=O)c1 c1(NC(C2N(C(=O)OC(C)(C)C)CCOCC2)=O)ccc(Cl)c2cn[nH]c12 c1(C(=O)NC2C3(CN(C(C(CC)SC)=O)C3)CC2)ccc(F)c(C)c1Cl C#CC1CN(C(c2ccc(C)c(F)c2F)=O)CCN1C(=O)C(C)O c1(NC(C)C)cccc([N+](=O)[O-])c1Br.N1S(=O)(=O)NC(=O)C1 C(C(COC)CC(=O)NC1(C(=O)N(CCCCOC)C)CC1(C)C)OC C(CCCCC(=O)NCC1CC(NC(c2cc(C(F)F)[nH]n2)=O)C1)OCC Cc1cc(C(=O)NCC(C2CCC2)NC(C23CSCC2C3)=O)ncc1F c1(CNC(c2ccc(CCC)[nH]2)=O)cccc(C(=O)NC2(C)CCSC2)n1 Cc1cc(C(C)C(N2CC(NC(=O)CC3CSC3)C(C)C2)=O)cc(F)c1 c1(CN(C(=O)CC2CCN2C(=O)CC2CCCC2)C)cc(Cl)ccn1 CCS(=O)(=O)CC(=O)NC1(C(=O)NC(c2ccc(O)nc2)C)CSC1 CCC(C)C(O)C(=O)NCC1CCC(NC(=O)CC2C=CCCC2)C1 O=C1CC(C(N2CCOCC2C(=O)NCCN2CCOCC2)=O)C2(CCC2)C1 N1(C(C(COC)CC(C)C)=O)CC2(CCCC(CNC(=O)CCCC3CC3)O2)C1 C1(n2cc(C(C)(C)CO)nn2)CC12CCN(C(c1ccc(F)s1)=O)CC2 Cc1cc(C)cc(C=CC(=O)NCCC(C)NC(C2CCC(=O)C2)=O)c1 c1(NCc2ccc(C)s2)ccnc(C(=O)NC(c2cnn(C)c2)C)c1 CCC(C)CCCC(=O)NCC1(F)CC(NC(=O)C(C)c2cccs2)C1 C1(CC(N2C(C(C)NC(=O)CCc3ccc(Cl)s3)CCC2)=O)CC2(CCC2)CO1 C1(C(=O)NC(C(=O)OC)C(C)O)C2CC(O)C(C2)N1C(c1ccc([N+](=O)[O-])o1)=O Cc1nn(C)c(N)c1NC(=O)NC(C)C(N1CCCC(N2CC(O)C2)C1)=O CC(O)CCN=C(NCCc1cccs1)NC1Cc2ccccc21 C1(NC(c2c(C)nco2)=O)CCC(C)(CNC(c2cc(F)n[nH]2)=O)C1 N1(Cc2c(C)n[nH]c2)CCC2(CC1)CC(NC(c1ncccc1Cl)=O)CO2 CC(CC(F)(F)F)C(=O)N1CCOCC(NC(c2cc(Cl)ncc2F)=O)C1 C(=O)(C1CCCc2cncn21)NCC#CCNC(C(=O)Nc1ccc(C)cc1)=O C1(NC(=O)C=C2CC2)CN(C(=O)Cc2cccc(F)c2)CC1C(F)F c1(C(=O)NC(C)C(CO)NC(=O)C(C)(C)N(C)C)ccc(C2(C#N)CC2)cc1 CC(C)(C)C(=O)C(=O)N1CC(CNC(=O)CCc2cccc(F)c2)C2CC2C1 C1(CC(=O)N(C2CCN(C(c3ns[nH]c3=O)=O)C2)CC)C=NN(C)C1=O N1(C(CCS(C)=O)=O)CCC(F)(F)C(CNC(c2cc(C(F)F)cs2)=O)C1 N1(C(C2(C)CC2Br)=O)CCOC2(CCN(C(C3CC4CC(=O)C3C4)=O)CC2)C1 C1(NC(c2cnc(C3CC3)o2)=O)CCN(C(C23CCCCC2C3)=O)CC12CCC2 CCC1CCC(=O)N1.C(C(CO)OC)NC(=O)COCCCOC N1(C(C2CCCC(NC(c3occc3Br)=O)C2)=O)CCc2n[nH]cc2C1 C1(C(NC(=NCC)NC2CCN(c3ccn(C)n3)C2)=O)CCC(=O)N(CC)C1 C1(F)(CO)CCCN(c2nccc(-c3c(Cl)cccc3Cl)n2)C1 c1(N2C(C)CCN(C(=O)CCN3CCCC3=O)CC2)ncnc2ccccc12 c1(C(=O)NCC2(C)CN(C(CS(N3CCN(C)CC3)(=O)=O)=O)C2)c(Cl)cccc1Cl c1(CCC)c[nH]c2ccc(Cl)cc12.Clc1ncccc1C(N1CCOCC1)C1CC1 CC1CC(NC(=O)C=Cc2ccc(C(N)=O)o2)CCN1C(c1cnnc(Cl)c1)=O c1(OCC(=O)NC(CNC(CCC2C(C)=NNC2=O)=O)C)c(C)cc(Cl)cc1Cl CC(C(CO)NC(c1csc(-c2cn[nH]c2)n1)=O)NC(C1CNC(=O)C1)=O c1(C(C)C)ccccc1NC(N(CCC(F)(F)F)CCC#N)=O C1(C(N(CC(C)NC(C=COCC)=O)C)=O)CCN(C2CC2)S1(=O)=O C1(NC(c2c(CC)csc2)=O)(CNC(=O)C(C#N)C(C)C)CC2CCC1CC2 Cc1cc(C)c(NC(=S)NCCc2ccc(C(c3ccccc3)=O)cc2)c(Br)c1 C1(NC(C2(Br)C(C)C2C)=O)CN(C(=O)C2=NNC(=O)CC2)CC1C1CC1 CC(C(=O)N1CCC(O)(CNC(c2n[nH]c3c2COC3)=O)C1)C(C)(F)F C1(CNC(CN(CC#C)C(C2CC2F)=O)=O)CCCN1C(C)=O Cc1cc(C(=O)N(C)C(c2cn(CCOC3CCOC3)nn2)C)cc(C)c1N O=C1CC(NC(=O)C(Cc2ccoc2)NC(=O)COCc2nc[nH]n2)CN1 C1(C(=O)NCC2CN(C(C)=O)CC2O)CCC(S(N)(=O)=O)CC1 N1(C(Cn2c(C)cnc2)=O)CC2CCC1C1CN(C(=O)C(C)NC=O)CC21 c1(C(=O)NC2CC(NC(C(Cc3c(C)noc3C)C)=O)C2)cccc2c1NCC2 c1(C(=O)NC2C(CNC(CCC(=O)OC)=O)C2)cc2cc(F)c(F)cc2[nH]1 C1(CNC(C(C=C)O)=O)CCN(C(c2nnsc2C(F)F)=O)CCC1(F)F N1(C(=O)C2=NOCC2)CC(C(CN2CCN(C=O)CC2)=O)C2(CC2)C1.OCCl N1(C(C2C(OC(C)=O)C2)=O)CCCCC(C(N2CCC(C#N)CC2)=O)C1 N1(C(Cc2c(C#N)cccc2)=O)CC2CCN(C(c3cncnc3)=O)C2C1 N1(CC)CCC(NC(C2(CCCNC(=O)CC3C(=O)ON=C3C)CCC2)=O)CC1 C1(C(C)(C)C(=O)NCC(C)(O)C2(C)CC2)CCCN(C(C2CCCS2)=O)C1 C(C(C)(C)CCOC)NC(C(C)NC(C1CCN(CC)C1)=O)=O C1(NC(Cc2cccc(OCC)c2)=O)CCC2(CC1)CC(NC(=O)CO)C2 Cc1noc2ccc(NC(C3CN(Cc4cc(Br)ncc4F)CCS3)=O)cc12 N1(C(c2c(CNC(C(C)C)=O)cco2)=O)CCC2(CCOC2)C1 c1(C(N2CCC(CCN(C)C(C3C=CCCC3)=O)CC2)=O)cc(F)cc(F)c1 C1(NC(C(C2CC(F)(F)C2)OC)=O)COCC1N(C)C1CC1 N1(C(C2CCC(C)O2)=O)CCCC2(CCCN2C(c2cccc(O)c2F)=O)C1 N12CCOC(C1)C2.C1(c2nn[nH]n2)(C(=O)O)CCCOC1 CC1=C(C)CC(C(N2CCCC2(C)CCC(=O)NCCC(C)C(C)(C)C)=O)CC1 c1(SC)ncccc1C(N1CCSCC1C(=O)Nc1cccc(I)c1)=O c1(OC)ccc2c(NC(C3CC4CNC(C3)C4)=O)ccnc2c1 CC(=O)C(C)CC(C)C(=O)NCC(=O)NC(C)(C)CCCF c1(OC)c(C(=O)NCC2CCN(C(=O)CC(C)C(C)C)C23CC3)ccc(Cl)c1C C(CCCCCC(=O)N1CCC(CO)C(O)C1)NC(C(C)C1CCCO1)=O c1(CN2CCC(CC(N3CC4COCC4C3)=O)CC2)c(Cl)cc(Cl)cc1Cl C(CCC(C)(C)C(=O)N1CCCC(CC(=O)NCC(C)(C)C(C)C)CC1)OC N1(c2ccnc(NC(c3ccn(CCF)n3)C)n2)CCC2(C)C(F)(F)C2(C)C1 c1(CCC)cc(C(=O)N(C2CCN(C(=O)C(CC)N(C)C)C2)C)[nH]n1 c1(NCC)cncc(C(=O)NC(CC2CC2)C(=O)NC(C)CN=[N+]=[N-])c1 c1(CC)ccccc1COCCOC.C12CCC(C1)NC1(CCC1)CNC2=O c1(C(C(N2CC(C(C(=O)N(C(C)CSC)C)OC)C2)=O)O)ccc(F)cc1 C(C)(C(=O)NC(C)CCSC)N(C(COCC)=O)CC CCN=C(NC1CC1C)N1CCCC(OC)C1.C1(C)(C)C(=O)N1.OCC c1(C(C)OC)nc(CO)cs1.N1(C(=O)CC2CC3CC3C2)CC(C(C)=O)(C(=O)NC)C1 N1(C(C(C2CCCCC2)C)=O)CCCCC(NC(c2cc3ccsc3[nH]2)=O)C1 c1(C(=O)NCC2CC(C)N(C(c3ccoc3Br)=O)C2)cnc2ncccc2c1 C1(NC(=O)C=CC=C(Cl)Cl)CCOC(CNC(=O)C(F)(F)CC2CCCC2)C1 c1(C(N2CC3C(NC(CCCC#C)=O)(CC3)C2)=O)c(F)ccc2c1CCCN2 CN1CC=C(CC(=O)NCCC2(O)CCN(C(=O)Cc3ccn(C)n3)CC2)CC1 c1(CC)cccc(C(=O)NC2CCN(C(=O)C(COC)CC)C2(C)C)c1F C(=O)(CCC(C)(C)O)NCC(C1CCCC1)NC(c1cn(CC)nc1C)=O C(=O)(C(F)C(=O)NCC(C(=O)N1CCC(N2CC(O)C2)C1)N(C)C)OCC C1(C)(CNC(CNC(CCC)=O)=O)CN(C(=O)C(C)NC(=O)OC)C(C)(C)C1 C1(NC(C(CCC)OCC)=O)C#CCCCCC1.C1(=O)COCCN1 c1(CC(=O)N(C2CC2)CC2CCCN(C(C(CSC)O)=O)C2)ccc(F)cc1Cl n1(CC)ncnc1C(=O)N(C)CCNC(c1sccc1CN(C)C)=O c1(CC(=O)NCC2(NC(c3ncoc3Br)=O)CC2)ccc(F)c(F)c1 C#CCC(C(=O)N1CC(O)(c2cn(CCNC(c3occc3C)=O)nn2)C1)C1CC1 C1(NC(=O)CC2CC23CC3)CC2CCC(C1)N2C(C1(c2nc[nH]n2)CC1)=O N1(C(CC2C(CNC(CC3C(C)CCC3)=O)C2)=O)CCOCC1CO N1(C(C(C)=C2CC2)=O)CCC(CO)C(O)C1.C12CCOCC1C(=O)N2 N1(C(c2c(C)cnnc2)=O)CC2CCCC2(NC(=O)CN2CCCCCC2=O)C1 c1(C(=O)NC2CCC(C)NC2)cc2c([nH]1)CCC2 c1(C2C(c3cn(-c4ccsc4)nn3)C2)ccc2c(c1)OCO2 CC(C)C1=NOC(C(N2CC(c3cccnc3)C2)=O)C1 C(CC(=O)NC1CC1C(=O)NCCCNC(=O)CCOC)(C1=CCCC1)OC c1(C(=O)NC2C3CC(NC(C(C)=C4CCC4)=O)CC32)cc(C#N)ccc1C C(C1CC1)(C1CC1)=CC(=O)NCCCOCCN(C(=O)CN1CC2CC2C1)C C#Cc1cccc(C(=O)NC2CC(CCNC(=O)C(C(C)C)OC)C2)c1Cl N1(C(CC2CCN(C(=O)CC3CSCCO3)C2)=O)CCCC(F)(F)C1 c1(CC(N)C(=O)NCc2occc2CN2CCOCC2)ccc(Cl)nc1 CC(C)C(C)C(CNC(=O)Cc1ccccc1COC(F)(F)F)NC(=O)CO c1(CN(C(=O)C(C2CCN(C(=O)CCn3ccnc3)C2)F)C2CC2)cccnc1 Cc1sc(O)nc1C(=O)NC(C)C(C)NC(c1cc(Cl)c(Cl)s1)=O N1(C(CN(S(CC)(=O)=O)C)=O)CC2CC(NC(=O)CCNC(C)=O)C2C1 c1(CC)c(C(N2CCCC(NC(C3CCC3)=O)C2)=O)cnc2cc(O)nn12 C1(COC)(NC(=O)C(C)C(F)(F)F)CCN(C(=O)Cn2cc(Br)cn2)CC1 c1(C(C(=O)NCCC#N)N(C2COCCOC2)CC)cc2c(cc1OC)OCO2 c1(C(N2CC3N(C(C(C)N(C)C)=O)C(CC3)C2)=O)cc(Br)c2nccn2c1 Cc1cc(C(=O)N(C(C)CCNC(c2c[nH]c3cccnc23)=O)C)c(N)c(C)c1 Cc1cc(C(C)(C)C(=O)NCC2(NC(c3ccsc3)=O)CCCC2)ccc1F CC1CN2CCCC2CN1C(C1CCC2(CC2)N1C(=O)Cn1cncn1)=O c1(C(=O)NC2CCC(N(C(CC(C=C)(C)C)=O)C)C2)cccc(F)c1C#N C1(CNC(c2c(C(=O)OC)csc2)=O)CCCCN1C(c1[nH]cc(C)c1C)=O c1(C(=O)NC(C(C(=O)NCc2c(C)scn2)(C)C)C)cncc2[nH]ccc12 C(=O)(CC(CCC)N1CC2(C=CCO2)C1)OCCCC C1(NC(c2c(C(=O)Nc3cccc(OC)c3)cccc2)C)CCC2(CCNCC2)O1 c1(OC)ncnc(C)c1C(N1CCN(C(=O)C2=CCCC2C)C(C)C1)=O CC1(C)CC(C(=O)NCC(C)(C)CNC(=O)CSC(=N)N)CO1 c1(OC)c(NC(C2CCCNCC2)=O)cccc1[N+](=O)[O-] C1(CC)Cc2ccccc2CN1C(=O)CCNC1CC1c1ccsc1 N1(CC)CCOC(C(=O)NCC(CNC(=O)COCc2ccncc2)CO)C1 C1(C(=O)NCC2C(OC)CCC2)CC2(CC(NC(C3CC4(CCC4)CO3)=O)C2)C1 N1(C(c2c(CC)noc2)=O)CCOC2(CCC(NC(c3cnc(Cl)[nH]3)=O)CC2)C1 c1(CO)cc2cc(CNCCN3CCN(c4ccccc4)CC3)sc2s1 Cc1[nH]c(=N)nc(O)c1CC(=O)NCCC1C(C)CCCN1C(=O)C=CCF n1(CCC)nc(C)cc1C(=O)N(C(C)CN(C(=O)C(C(C)C)n1ccnc1)C)C c1(C(=O)NCC2(C)N(C(C(C)OCC3CC3)=O)CCC2)ccc2c(c1)CCO2 c1(CC(=O)OC(c2ccc(C)s2)c2ccco2)nnc2n1CCCC2 N1(C(C2(OC)CC2)=O)CCn2ncc(CNC(c3c(C)ncnc3C)=O)c2C1 CC1=C(C(=O)NC2CCC2NC(C2CC(CC3CC3)C2)=O)SCCO1 CC1=NNC(=O)C1CC(=O)NCCC1CCN(C(=O)C=Cc2ccncn2)C1 C1(CNC(N2CCC(c3ccc(CN(C)C)cc3)C2)=O)CCC(O)(C2CC2)CC1 c1(CNC(N(c2cc(Br)ccc2OCc2cccnc2)C)=O)ccc(F)c(Cl)c1 C(CNC(=O)C(C)n1ccnc1)(CC(F)(F)F)NC(c1c(C(C)C)nccc1)=O C(=O)(C1CCCn2ccnc21)NCC1CCN(C(C(CCC)(C)O)=O)CC1O c1(CNC(COCCCC)=O)ccc(CNC(c2ccc(C(C)=O)cc2)=O)cc1 C(CC(C)C)(C(=O)NCCN(CCOC)C(C1(C)CC1(Cl)Cl)=O)OC CC1C2CN(C3CCCN(C(=O)CC(=O)NC(C)(C)C)C3=O)CC12 C1(NC(CCc2ccn(C)c2)=O)CCC(C)(CN=c2[nH]ncs2)C1 Cc1cnc(N2CC(C)(c3nc(-c4cccs4)no3)C2)nc1 N1(CCOCCOC)CCC2(CCCCN(C(=O)CCN3CCCS3(=O)=O)C2)C1 C1(NC(CCCNC(N)=O)=O)CCC12CCN(C(c1cn(C(F)F)cn1)=O)CC2 c1(C(C(C)C)N)cn(C2CCCC2)cn1.c1(C(C2(C)CC2)C)nnnn1C(C)(C)C c1(CN2CCC(CCC)(CO)C(O)C2)cc2c(cc1C(=O)O)OCO2 N1(Cc2ncc(C)c(Br)c2)CC2C(C1C(=O)NCCc1ccsc1)C2(C)C c1(C(=O)NCC(C)(CO)NC(COCCC=C)=O)cccc(-c2ccco2)c1 c1(-c2n(C(COC)C)nc(Cc3ccccc3C)n2)ccc(OC)c(C)c1 C1(C(=O)NCC2(CCNC(C3ON=C(C)C3)=O)CC2)CCCCCC1 C1(CNC(Cc2cnc(C)s2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1 CCC(C)CCCCC(=O)NC1CC(NC(=O)CC(C)(C)C(=O)OCC)C1 C1(NC(CN2CCC(C)CC2)=O)CC2CCC(C1C)N2C(c1ccc(O)nc1)=O N1(C(CC(C)c2ccsc2)=O)CCC2(CC1)CC2CNC(C1C2CCC(=O)C12)=O C(C(COC)CC(=O)N1CCCC1CCNC(C1CN(C)C1)=O)OC N1(C(CC2C(C)C2)=O)CC2CC3CC2C1C3NC(C1C2CNC(=O)C12)=O N1(C(c2ccc(C(C)=O)[nH]2)=O)CCC(CCN(C(=O)COC2CCOC2)C)CC1 C(=O)(C(C#N)CC)N1C(C(=O)NCC(C#C)OC)C(C)C1 C(CN=c1[nH]c(=NCCN(CCCN(C)C)C)[nH]c2c1CSC2)c1c(C)nc[nH]1 C1(CC(N2C(C)CC(NC(CC(C)OC)=O)C2)=O)CCCCC1(C)C c1(C(N2C(CNC(CC3(OC)CC3)=O)CC3CC32)=O)nn(C)c2ccc(F)cc12 n1(CC(C)CO)nc(-c2ccn(C)n2)nc1-c1cnn(CC(F)(F)F)c1 c1(C(=O)OC)cnn2c1CN(c1cc(C)nc(O)n1)CC2 C(CCCC)(C(=O)N1CCCC1CCCC)NC(C(CC#C)O)=O C1(C(N2CCC(C#C)(O)C2)=O)CC(N=[N+]=[N-])CN1C(c1ccnnc1)=O C(C(C)N=c1[nH]nc(Cl)c(C)c1C#N)(C1CCCCC1)NC(C)=O C1(C)(CC)C=C(C(=O)NC(CNC(c2ccc(Cl)cc2Cl)=O)CO)C1 C1(C(=O)OC)CCC2(CC(C(N3CCOCC3CC(C)C)=O)C2)NC1 S(=O)(=O)(c1ccc(Br)cc1NCC1C2CCCOC12)NC(CC(C)(C)OC)C c1(NC(C2C(C(C)NC(C3CC3C(C)(C)C)=O)OCC2)=O)cncc(CO)c1 c1(C(=O)NCCN(C(=O)NC(=O)NC)C2CC2)ncc(C)cc1OC(F)F C=CCC(CC(F)F)C(=O)NCC1CCN(C(=O)Cc2ccc(C)nc2Cl)C1 CCCCC(C(=O)NCCCC1CCN(C(=O)C(O)CSC)CC1)N(C)C C1(CNC(C2(CSC)CCC2)=O)CC(O)CN1C(=O)CCCCN1CCCC1 C1(C(=O)NC2CN(C(c3c(F)ccc(C#N)c3)=O)C2)CC(c2ccncc2)=NO1 c1(C(=O)NC(C(c2scc(C)n2)C)=O)cc(O)nc(C(F)F)n1 C1(=CC(=O)NCCC2(OC)CN(C(=O)CCc3cnn(C)c3)C2)CCN(C)CC1 C1(F)(CNC(c2ccco2)=O)COCCN(C(C2(CF)CC(F)(F)C2)=O)C1 C(=O)(CCC(F)(F)C(=O)N1CCC(NC(=O)CC(CC)CCCC)C1)OCC C1(NC(c2nc(C#C)sc2)=O)CN(C(c2ccc(C)nc2O)=O)C(C)(C)C1 c1(NC2C=CC(C(=O)OC)C2)cccnc1NC(C=CCOCCOC)=O.C(C)(C)O N1(C(CC(C)OC)=O)CCCC(C2CCCN(c3cc(Cl)ncn3)C2)C1 C1(C(N2CCN(c3ccc(Cl)nn3)CC2)=O)CCCN(c2ccc(F)cc2)C1=O N1(C(=O)C=CC=C(Cl)Cl)CCN2CCN(C(=O)CCC(=O)c3ccccc3)CC2C1 C1(NC(C(CC(C)C)O)=O)CN(C(C2(C)CCOCC2)=O)CC12CCC2 C(=O)(CS(=O)(=O)C1CC1)NC1C2CC(NC(COCCOC)=O)CC21 C1(C(=O)NCC23CCCC2C3)CCOCCN1C(=O)CCCc1cnn[nH]1 c1(C(N2CCC3(C(CNC(=O)CC(F)F)C3)CC2)=O)cc2ccc(Cl)cc2[nH]1 c1(NC(CCCC(C)C)C)nc2ccccc2[nH]c1=NC1CCn2ccnc2C1 N1(C(c2n(CCC)ccc2)=O)CCC(C)(C)C1CC(=O)N(CC(F)(F)CO)C C(C)(C(=O)NC1CC(NC(C2(c3ccc(Cl)nc3)CCC2)=O)C1)(C(C)C)OC CCCCCC(CC)C(=O)NC(CC1CC1)C(=O)NCc1cccc(C2CC2)c1 C1(NC(C2CCn3c(Br)cnc3C2)=O)CN(C(=O)C2CC2)C2(CCCC2)C1 C(=O)(NN1CCCC1C(=O)OC)C1(C)N(C(CC=C)CC(F)F)CC(O)C1 N1(C(C2N(C(C3CCC(C)(C)C3)=O)CC(O)C2)=O)CCc2nncn2CC1 c1(OCC(=O)NCC(CCNC(c2cncc(C)c2)=O)O)cccc(Cl)c1Cl c1(C(=O)NC(CN(C(=O)CCC2NC(=O)NC2=O)CC)C)coc(S(N)(=O)=O)c1 CCC(O)C(F)(F)C(=O)N1CCC(C)(NC(c2ccn(C3CC3)c2C)=O)CC1 c1(C(N2CC(N(C(C3CCN(C(C)=O)CC3)=O)C)C(F)C2)=O)ccc(=O)n(C)c1 C(C1Cc2ccccc21)NC(C(CC1CC1)NC(c1cncc(C)n1)=O)=O N1(C(C2C(=C)C2)=O)CCCC(CO)(NC(c2cccnc2NC(C)C)=O)C1 C(=O)(C1=CS(=O)CCC1)N1CCC(C)(NC(=O)CC=Cc2ccccc2)CC1 N1(C(C(C2CCCC2)OCC)=O)CCOCC1CNC(C1CCCC1)=O c1(C(N2C(CC)CCC2C)=O)coc2c1CN(C(C1CC3(CC3)CO1)=O)C2 CC(C(C)(C)NC(c1cnc(-c2ccoc2)s1)=O)NC(c1cc(C(F)F)on1)=O c1(CCNC(=O)CCN(C(=O)CC2CCSCC2)C2CC2)ccc(F)cc1 C1(C(N2CCN(C(C(CC(C)C)(C)C)=O)CC2C)=O)CCC2(CCOCC2)O1 c1(C(N2C(COC)CN(Cc3cn(C)nc3C)CC2)=O)cccc2c1OCO2 Cc1ccc2c(C(=O)NC(CNC(=O)C(C)CC3CCC3)C3CC3)coc2c1 C1(CC)CN(C(C2CCCC23CC3)=O)CCCN1C(=O)Cc1cccc(Cl)c1F c1(NC(=O)NCC2(OCCSC)CCCC2)cc(CC(C)C)nc(O)c1 C1(CNC(CC=C)=O)(OC)CCN(C(C2CCN(CCCC(C)C)CC2)=O)CC1 Cc1cc(-c2cn(CC3CCN3C(C3(C(N)=O)CC3)=O)nn2)cc(C#N)c1 c1(NC(CC)CNC(=O)C2=NOCC2)ncnc2cc(C)[nH]c12 c1(OCC)c(C)ccc(NC(c2nnnn2C)c2csnn2)c1C CC1(CNC(=O)CN2CCC(O)CC2)CCC(NC(=O)CNC(=O)C2CC2)CC1 CCC(CC(=O)NC(C1CCCN1C(=O)C(CSC)OC)C)C(C)C N1(C(COC)=O)CCCC12CCN(C(C1CC(F)(CO)C1)=O)C2 N1(C(C2N(C(CCC)=O)CSC2)=O)CCC(C)(NC(=O)CSCC(=O)OC)C1 N1(C(c2c(CC)n(C)nc2)=O)CC(NC(=O)Cc2ccco2)CC12CCCOC2 N1(C(c2cc(C)no2)=O)CCC2(CC1)CC(C)N(C(=O)C(F)C1CC1)C2 c1(C(=O)NCC(C)(CO)NC(C(CSC)O)=O)cnn(C2CC2)c1C N1(C(c2ccc(COC)s2)=O)CCN(C(=O)CS(=O)(=O)NC)CC1C1CC1 N1(C(CCOc2c(OC)cccc2)=O)CC(CNC(C2CC2F)=O)CC12CCC2 N#CC1(C(N2CCC(O)(CNC(=O)C=Cc3cncc(F)c3)C2)=O)CCCCC1 C=CCCC(O)CN(C(=O)C(c1ccccc1)NC(C1(CO)CC(C)(C)C1)=O)C c1(OC)ccc(C)cc1CN1CCC(NC(C2(C3CCCO3)CC2)=O)C(C)C1 c1(SC)ccccc1NC(c1cc(F)ccn1)c1nnnn1C1COC1 C#Cc1ccc(C)c(NC(C2CC(C)N2C(=O)C(C)(C)n2cnnn2)=O)c1 c1(OCC)cccc(CC(=O)NC2CCCC2CNC(c2nc(C)sc2C)=O)n1 N1(C(c2ccc(C)o2)=O)CC(CNC(c2occc2Br)=O)C2(CC2)C1 n1(CC(=O)NCC(C)N(C(c2cc(SCC)ncc2)=O)C)nc(C)c(Br)c1C CC(C)CC(=O)NC(C)(CNC(=O)CCCONC(=O)OCC(C)(C)C)CO c1(C(C)NC(c2cccc(F)c2I)C(=O)OC)ccc(Br)cc1OC c1(C(N2CC(C)C(CNC(C3CC(=O)CCO3)=O)CC2)=O)ccc2ncsc2c1 Cc1ccc(F)c(C(N2CCN(C(C3CN(C)CC3(C)C)=O)CC2)=O)c1O Cc1cc(F)ccc1C(=O)NC1CCN(C(=O)C(C)OCC(F)(F)F)C1C(C)C C(=O)(C(C(=O)N(CCCN(C)C(c1ccccc1C(N)=O)=O)C)OC)OC CC1CCN(C(=O)CCCNc2ccccc2)CC1CNc1nnccc1C#N C(=O)(C1CCCc2cccnc21)NCCC(C)NC(Cc1c(C)cc(O)cc1)=O CCC(C)(CNC(c1cc(F)ccc1C)=O)C(=O)NC(CC(C)C)C(N)=O c1(C(=O)NC(C)C(C)NC(C2CCC2)=O)cc(Br)cn2ccnc12 C#CC(CNC(C1(NC(c2csc(C#N)c2)=O)CCCC1)=O)CC(C)(C)C C=CCC(F)(F)C(=O)NC(C)CN(c1cc(O)nc(SC)n1)C c1(OCOC)cc(CNCc2cccc(-c3ccco3)c2)cc(N)c1OC C1(C(=O)NCC(C)NC(C(C(C)C)SCc2ccccc2)=O)CC2(CCC2)CO1 CCC(O)C(C)(C)C(=O)NCC(C)(C)CC(=O)NCCCc1nc(C)no1 Cc1cc(C)nc(SCC(N2CCN(C(C3C4COCC34)=O)C(CO)C2)=O)n1 c1(OCC(=O)NC2(CC=C)CN(C(=O)C=C(Cl)Cl)C2)ccc2c(c1)CCC2 C1(NC(c2c(C)onc2CO)=O)CCC2CN(C(C3COC(C)C3)=O)CCC2C1 C(CCC)(C(=O)NCC1CCCCC1C(=O)NCC1CCC2(CC2)C1)=CCC N1(C(c2cnc(OC)s2)=O)CC(C(=O)NC(C)CC(C)C)C(C)(C)C1 N1(C(c2cc(C)oc2)=O)CC(O)(C2(CNC(=O)C(C#N)C(C)C)CC2)C1 C1(=O)CCCC(CC)N1.c1(CCC)ncc(C(=O)NC2(C#N)CCC2)cn1 C1(NC(C=Cc2ccc(OC)c(C)c2)=O)CN(c2nnco2)C2(CCOCC2)C1 Cc1c(C(N2CCC(O)(CNC(C3(Cl)CC3)=O)C2)=O)cnn1CCN(C)C C(C)(C(=O)N(CCCNC(=O)CCC1CC1(C)C)CC1CCCC1)=C(CC)C c1(C(N2CCC2C2CCC2)=O)cccc(Cl)c1.C1(=O)C(C2CC2)C2C(C2)CN1 Cc1cc(C)c(C=CC(N2CCC2CNC(C2(C3(O)COC3)CC2)=O)=O)c(C)c1 C1(SCCCNC(c2cnoc2-c2ccccc2)=O)CC=CCC1 C1(NC(c2cc(C)n(C(F)F)n2)=O)CN(C(c2cccc(CF)c2)=O)C(C)(C)C1 C(C(=O)N=c1ccn(-c2ccc(C)cn2)[nH]1)=C(C)Cc1c[nH]ccc1=O C1(NC(C=C(C)C(C)(C)C)=O)CN(C(=O)CCCCC2CCC2)C2(CCOC2)C1 C(=O)(C1=NNC(=O)CC1)N1C(CN(C(c2cn3c(n2)CCC3)=O)CC)CCC1 c1(C(N(CCCN(C(C2CCC(C)C2)=O)C)C)=O)cc2nccnc2cc1F CC(C(F)C(=O)NC1CCC(N(C)C(c2cnc(S)[nH]2)=O)CC1)C(F)(F)F C(CC(CNC(=O)CCc1ccsc1Br)NC(=O)COCCF)OC c1(OC)ccc(NC(=O)C(F)C(C)CNC(=O)CSc2nc[nH]n2)c(O)c1 c1ccc2nc(N3CCC(CN4CCCC4)CC3)ncc2c1 c1(C(OCOC)C)ccc(C(=O)C(C)=O)o1.C(=O)(C(C)C)N(C(=O)CO)CC C1(CNC(=O)NCCc2cc(F)c(Br)cc2Cl)C2Cc3cc(F)ccc3C12 Cc1nccc(C(N2CC(NC(=O)Cc3ccnc(Br)c3)C(C)(C)C2)=O)c1C N1(C(=O)NCC(C#C)CC(C)C)CC2OC(=O)N(CC3CC34CC4)C2C1 c1(C(=O)NC)cc([N+](=O)[O-])ccc1N(CC(C)NC(=O)C(C)(C)SC)C C(C(C)(C)CC(=O)N1CCOCC1CN(C(=O)C(N1CCN(C)CC1)C)C)OC C1(NC(C(N2CCSCC2)C)=O)COCCN(C(=O)CCOC2CC2)C1 C12(CC(=O)Nc3cnc(Cl)cc3Br)CCC1CN(Cc1cc(Br)cs1)C2 c1(OC)c[nH]nc1C(=O)NCC(C1CC1)N(C)C(c1sccc1OC)=O C(=O)(C(C)(C)C(F)F)NCC(C1CN(C(=O)C#CC2CC2)CCO1)(C)C c1(C(=O)Nc2c(CC)nc(Cl)cn2)ccc2c(c1)CCC(=O)N2 C#CC1(O)CC(C(N2CCC(C(=O)N(C)CC3(O)CCOC3)C2C)=O)C1 CC1CC(C(=O)NCC(C)(O)CN(C)C)N(C(=O)C(O)CN2CCCC2)C1 CCC(C(=O)NC1(C)CC(NC(=O)Cn2ccccc2=O)C1)C(C)(F)F C#Cc1cncc(C(N2CC(CNC(=O)C=C(CC)CC)CC2(C)C)=O)c1 CC#CCC(C(=O)N(C)CC1(CO)CC1)NC(c1c[nH]c2cnccc12)=O c1(C(=O)NCC2CCC(NC(CC(C)n3cccn3)=O)C2)ccc(F)c(C#N)c1 c1(C(=O)NC(CNC(Cc2cn(CC)nc2)=O)C)ccc(OC(F)F)nc1 c1(NC(C2C(CNC(c3cc(C4CC4)no3)=O)CCC2)=O)ccc(CCO)cc1 N1(C(Cn2ncn(C)c2=O)=O)CC=C(CCNC(C2COCCO2)=O)CC1 C(c1ccc(Cl)cc1F)=CC(=O)NC.C(=O)(NCC)NCCN1CC1 CC(C)C1=NOC(C(=O)NCCCC(=O)NCC=CCl)C1 C(N=c1nc2c(c[nH]1)nc(N1CCC3(CCOCC3)C1)n2C)C1CCC(C)C1 N1(C(C(CC)C(F)(F)F)=O)CCOC2CN(C(=O)Cn3nccc3C)CC12 C1(OC(C)(C)C)CCC2(CC1)CC2NC(c1snc(C)c1C(=O)O)=O.C(=O)(N)O Cc1cc[nH]c(=N)c1C(=O)NCC1(F)CC(CNC(=O)C(O)c2ccsc2)C1 c1(C(C)C(=O)N(C)CC2CCCCN2C(=O)CCC(F)F)cc2ccccc2s1 C1(O)(CNC(CN(C(=O)COC2CCOCC2)C)=O)CCOCC1 N(C(=NCCCCl)NCc1ccc(C(N)=O)o1)C1C(C)(C)C1 C1(NC(C=C(CCC)CCC)=O)CCCN(C(=O)C(C)OC2COC2)CC1 c1(C(=O)NCC2C(CNC(Cn3ncc(C)c3)=O)C2)ccc(C2CC2)cc1 CC1CCCN(C(=O)C(=O)NC2C3CC2N(C(=O)CSc2ccccc2)C3)C1 C1(NC(c2c(C(C)C)cco2)=O)COCCN(C(=O)C(C)n2cccn2)C1 Cc1n[nH]c(C)c1C(C(C)C)NC(=O)NCCCC(=O)NC1CCCOC1.OC c1(C(CNC(C2CCCN2C(N)=O)=O)OC)c(F)cccc1F.C1(C(=O)N)CCC1 c1(C(N(CC(C)NC(=O)C(F)n2ccnc2)C)=O)cc2c(O)cc(Cl)cc2[nH]1 Cc1ncc(C)c(=NCC(C)NC(c2ccc3nc(O)[nH]c3c2)=O)[nH]1 N1(C(CN(C(=O)CC2CC(NC(C)(C)C)C2)C(C)C)=O)CCc2ncsc2C1 N1(C(C=CC=CCC)=O)CC2CCCC2(CNC(=O)CCc2cncs2)C1 N1(C(CN(CCOC)C(c2nonc2C)=O)=O)CCC12CCN(C)C2 c1(C(=O)NC23CC(NCc4cncc(Cl)c4Cl)(C2)C3)ccc2ncnn2c1 C123CCC(CC1)(C2)OC3.Cc1cc(CNC(N(C)Cc2ccccc2)=O)on1 c1(C(=O)NCC23CC2CN(C(c2cc(Cl)no2)=O)C3)cn2ccccc2n1 C=CCCCCCCCCC(C)(C)C(=O)NCC(C)(C)NC(C1CC(C)=NO1)=O c1(C(=O)NCC(CC)NC(=O)NC(C)C)sc(C(C)C)nc1C n1(CCC(N2CC(NC(=O)CCC(F)(F)F)C(O)C2)=O)ccc2ccccc12 Cc1csc(NC(=O)C=Cc2ccc(Br)cc2)c1C#N.c12cncc(c1)S2 N1(C(C2CCCN(C(C)=O)C2)=O)CCCC(O)(CNCC=C(C)C)C1 C1(CCC=C)CN(C(c2ncccn2)=O)CCN1C(=O)CC(=O)OCCC Cc1cccc(C(=O)NC2CN(C(c3cnc(C4CCCO4)s3)=O)CC2C)c1O c1(C(=O)Nc2c(C)nc(NC3CC3)s2)[nH]nc2c(=O)n(C)cnc12.C(C)(COC)S C12(NC(c3cnc4sccn34)=O)CCCC1N(c1ccnc(C(F)(F)F)n1)CC2 C=CC1(CC(=O)NCC2(O)CCOC2C)CN(C(c2ccc[n+]([O-])c2)=O)C1 C1(CNC(=O)Cc2cccc(Cl)c2)CN(c2ncncc2Cl)CCCO1 C1(C(N2C(CN(C)C)C=CC2)=O)CC(=O)CN1C(c1ccncc1)=O c1(C(=O)NCC2(C(=O)N(C3CC3)Cc3nc[nH]n3)CCCO2)cccc2c1CCC2 Cn1ncc(CNC(c2cc(C(N)=O)[nH]n2)=O)c1C(=O)NCC1(O)CCCOC1 c1(OC)ccc(C(CNC(=O)CO)NC(=O)CCC2CCN(C)C2)cc1 CC1(C(=O)NC2CCCCC2NC(c2cncc(O)c2Cl)=O)CCC(=O)NC1 C(c1cccnc1)=CC(=O)N(C1CN(C(=O)CN2CSCC2=O)C1)C C(C(CC(C)C)C(=O)NCc1cccnc1C(=O)NC(c1cnc[nH]1)C)OC c1(C(=O)NCCN(CC(C)O)C(=O)C=C(C2CC2)C2CC2)cccc(N)c1F C1(CNC(c2n(CC)nnn2)(C)COC(C)C)CCSC1(C)C c1(CC(C(C)C)Sc2ccsc2)cccc(F)c1.C1(=O)NO1 N1(C(C(Cc2ccccc2)OC)=O)CCCCC1CNC(C1CCCCN1C)=O C1(CNC(C)=O)CCCC2(CN(C(c3cccn(O)c3=O)=O)C2)O1 C(=O)(C1COc2ccccc21)N1CC(NC(c2scc(OC)c2)=O)CC2(C1)CC2 Cc1cccc(C(N2CC(O)CC2CNC(=O)CCn2ccnc2)=O)c1 C1(C(=O)NC(C)C(C)NC(c2ccc(N)cc2Cl)=O)(OCC)CCC(F)(F)CC1 c1(C(=O)NC2C(CNC(=O)C=CCN3CCSCC3)COC2)cccc(O)c1F N1(C(C(C)OCC=C)=O)CCC2(C1)CN(C(C1CCn3nccc3C1)=O)C2 C1(CC(=O)N(CCCNC(CC(C)C)=O)C)CCC(C)(C)O1 CC(C)(F)CCC(=O)NC1(CF)CCN(C(=O)CONC(=O)OC(C)(C)C)C1 C1(CNC(c2cccnc2F)=O)CC(N=c2[nH]c(Cl)ncc2Cl)C1 C1(CCNC(C(CC)(C)CC)=O)CC2CCC(C1)N2C(C1CNC(=O)N1)=O C1(CCCCCNC(C(c2cnn(C)c2)C)=O)CCN(C(C2(C)COC2)=O)CC1 C1(C(=O)NCC2CCN(C(=O)CC=C(Cl)Cl)C2)C2C3CC4C1C1C2CC3C41 N1(C(CCCC)=O)CC(NC(c2cc3sc(C)cc3s2)=O)CC12CCCC2 c1(OC)cccc2cc(C(=O)NC(CCNC(=O)C(C)NC(C)=O)C(C)C)[nH]c12 CC1(C)CCCCC1CC(N1CC2CC2(NC(c2coc(CO)c2)=O)C1)=O c1(C(CCC(=O)OC)NC(c2ccoc2)CC)cc(C2CCC2)on1 CCC(CNC(=O)C(CNC(c1cnn(C)n1)=O)CC1CC1)CCO CC1(C)OC(=O)NC1C(=O)NCC(CNC(=O)CCn1ccccc1=O)CO C(=O)(C#CC1CCOCC1)N1C(CCCNC(C=CC=CCC)=O)CCCC1 N1(C(c2c(C#N)cccc2Cl)=O)CCCC2(CCC(NC(=O)COCCF)C2)C1 c1(CCNC(N2CCC(n3cnnc3)CC2)=O)cc2ccccc2s1 CCC(C)(C)CC(=O)NCC1CN(C(c2nnn(C(C)(C)C)n2)=O)CCC1C CCCCCCC(C)c1nc(-c2ccc(OC)nc2)nn1-c1ccnc(Cl)c1 C1(C(N2C(CNC(c3cc(F)c[nH]3)=O)CC(OC)C2)=O)CCCC2(CC2)C1 C1(CC)CCCC(CNC(C2C=CC(NC(c3coc(N(C)C)n3)=O)C2)=O)C1 C1(NC(c2ccc(CC)[nH]2)=O)CC1C1CCCN(C(C23CC2COC3(C)C)=O)C1 c1(C(=O)OC)ccc2c(c1)CC(NC1CCC3(CC1)CN(c1nnnn1C)C3)C2 C1(C(=O)NC2CC3(CN(C(CNC(C)=O)=O)C3)C2)COc2ccc(F)cc2C1 CCN=c1ccc(C(=O)NCC2CCN(C(=O)C(O)C3CCCC3)C(C)C2)c[nH]1 c1(CNC(=O)C(N2CC(O)CC2c2ccc(F)cc2)C2COC2)ccccc1Br N1(C(c2c(C#N)cn[nH]2)=O)CC2CCCC(C1)N2C(c1ncccc1Cl)=O C1(CC(=O)N(C)CCNC(c2ccc(C(F)(F)F)o2)=O)CC(O)C1(C)C C1(F)(CNC(c2cc(CC)[nH]n2)=O)CCC(CNC(=O)C=CC2CCC2)C1 CC(C)C(C(=O)NC1CCCC1NC(c1ncoc1C1CCC1)=O)NS(C)(=O)=O N1(CC)CCCN(C(=O)C(C2CC=CCC2)NC(c2onc(C)c2CC)=O)CC1 c1(CCC(=O)NC2CCC(NC(CCOCCN(C)C)=O)C2)cccc(F)c1F C(=O)(C(C)(C)CCCNC(=O)CC(C)C)N(CCCC)CCCO c1(C(N(C2CCCN(C(=O)CN3CCCC3)C2)C)=O)cccc(-n2cncn2)c1 CC(C)C(CCC(=O)NCc1c[nH]c2ccccc12)NC(C1C=CCS1)=O c1(CNC(N(CCC=C)CC)=O)ccc(CCCC#N)cc1 C=CCCCCC(=O)Nc1cccc(CNC(c2n[nH]cc2C(C)(C)C)=O)c1 C1(C(N2CC(O)(C3CCCN3C(=O)C=CC3CCC3)C2)=O)(CC)CCNC1=O c1(CNC(c2c(CC)ocn2)=O)ccccc1CNC(c1ccn(CCF)n1)=O c1(CC)ccc(C(N2CCCC(NC(=O)C(C)(O)C3CC3)C2)=O)cc1Cl N1(C(C2(SC)CC2)=O)CC2C(CNC(=O)C(N3CCSCC3)C)C2C1 c1(CC)cccc(C(N2CCC(O)(CNC(c3ccnnc3S)=O)C2)=O)c1F CCC(CN(C)C)CC(=O)N1CCC(C(N2CC3CC(C)C3C2)=O)CC1 C(=O)(C1=NOC2COCC12)NC1(C(N2C(COC)CC2)=O)CC1(C)C C1(CC(F)(F)F)C(=O)N1.c1(CNC(=O)COC(F)F)cccc(C(F)(F)F)c1 C1(NC(C2(COC)CC2)=O)CN(C(=O)COc2cccc(Br)c2)C2CC12 c1(CN2C(C(=O)NC3CC=CCC3CO)CCC2)c(Cl)cccc1Cl Cc1cc(C(N2CCC(C)C(NC(c3ncccc3F)=O)C2)=O)c(O)nc1C C1(NC(C2C(=C)CC2)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)CC1F CCC(CC(=O)N1CC2(C)CC1(C(=O)NCC1CCC(CO)O1)C2)C(C)(C)C N1(C(CNC(=O)OC)=O)CCN(C(=O)CC(F)(F)C(C)(F)F)C(C)CC1C C(=O)(C(F)(CNC(=O)Cn1c(C)ccc1C)C(C)C)N1C(C=C)CC1 c1(CC)[nH]nc(C(=O)NC23CC(C2)N(C(c2ccccc2C(C)=O)=O)C3)c1C C1(C(C)NC(Cc2nc(C)oc2)=O)CCN(C(=O)Cn2ccc(Br)n2)CC1 C(CCC(=O)NCC1C=CCN1C(=O)COC1CCOCC1)N(C)C c1(SC)cccc(C(=O)NCCC(O)CNC(=O)COc2ccsc2)c1 c1(C(=O)NCC2CC(C)N(C(=O)CC(C)(C)C(F)F)C2)cn(C)c(=O)n(C)c1=O N1(C(COCC#C)=O)CCN(C(c2ccc(C)c(C)c2)=O)CC1C1CC1 c1(C(N2CC(O)(CCNC(C(CC)N(CC)CC)=O)C2)=O)cccnc1S N1(C(c2c(C)nn(C)c2Cl)=O)CCC(C)(C)C(NC(c2occc2Cl)=O)C1 C(=O)(CCCS(N)(=O)=O)N1CC(C)(CNC(=O)C#CC2CC2)OCC1 C1(CC)C(=O)N(C)CCN1C(=O)C(C)(CSC)NC(C1CC2(CC2)C1)=O c1(C(=O)NC(CCCCNC(CCC(C)OCC)=O)C)cc(C)nc(O)c1 C(C(CC(C)(C)C)C(=O)O)NC(CC1CC(CC)OCC1)=O N1(CCN(C)Cc2cc(CC)n[nH]2)CC2(CC2C(=O)OC)C1 c1(C(=O)NCC(CC)NC(=O)CC2(C)CC2)c(C)ccc2nsnc12 N1(C(C(C)(C)OCC)=O)CC2C3CCC(C2C1)N(C(=O)CCc1ccccc1)C3 N1(C(C(CC=CC)C)=O)CCOCC(C(=O)NCCCCCCCO)C1 c1(C(C)NC(=O)CC=CC(=O)N(C)C)ccc(OC(=O)C(C)(C)n2cnnn2)cc1 c1(C(=O)NCC2CC3N(C(C(C)=CC)=O)C(CC3)C2)c(F)ccc2n[nH]cc12 N1(C(CCSCCCC)=O)CC(NC(C23C4CC(CC24)C3(F)F)=O)CC(C)(C)C1 N1(C(c2cccn2-c2ccccc2)=O)CC2CCC1C(NC(C13CC(C1)C3)=O)C2 N1(C(c2ccc(C3CC3)o2)=O)CCOC2(C1)CN(C(=O)C(F)(F)C1CC1)C2 C(=O)(CC(O)CC(C)C)NCC1(c2ccccc2)CCN(C(C(C=C)CC)=O)C1 c1(C(=O)NC2CC(F)(CNC(C3C(=C)C3)=O)C2)ccc(SC(C)C)cc1 C(=O)(C1=CCC2CCC1N2C(c1nc(O)sc1C)=O)NCCN(C)CC c1(C(=O)NCCN(C(=O)Cn2cc(Br)cn2)CC)ccc2c(c1)N(C)C(=O)CC2 c1(OC)ccc(CN2CCC(C(=O)NC(c3ccccc3)C)C2)cc1C c1(CC=C)ccccc1C(=O)NC(C(=O)NC1CCCC1CCOC)C(C)OC C=C(C)C(C)(C)C(=O)N1CCC1CC(=O)NCC1(COC(C)=O)CC=CC1 c1(NCc2n(C)nnc2)nc2ccccc2nc1NCC1CCCCS1(=O)=O N1(C(=O)Cn2cc(C3CC3)cn2)CCN(C(=O)Cc2nncs2)C2CCCCC12 C=CCC(CC(=O)NC1(C)CCOC1C)NC(c1cc(=O)n(C)cn1)=O c1(C(=O)N)ccc(SS)cc1C.C1(c2cn(CC3(CC)CC3)nn2)C(C)(C)C1(C)C N1(CCCC)CCCCC1C(=O)NCC(CO)NC(c1ncsc1C1CC1)=O C(CCC(C)C)(C(=O)NC(C)CCSC)NC(C(C)(C)OCCC)=O CN1CCC(C)(C(N2CCC(C)(CNC(c3cnc(O)o3)=O)C2)=O)C1=O CCCCC(CC(=O)N1CCCCC1CC)NC(C1CCN(CC)C1C)=O C12(CC(N3CC4(C3)CN(C(C35CCCCC3C5)=O)C4)=O)CNC(=O)C(C1)C2 C1(C(N2CCC(O)(CNC(c3cc(=O)cc[nH]3)=O)C2)=O)CCC2(CCC2)CO1 C1(NC(C=C(C)C(C)C)=O)CC(NC(c2cncc(N)c2)=O)C12CCC2 c1(C(=O)NC(CN(C(C(C)OCCCCCC)=O)CC)C)cnc(C)n1C(F)F Cc1cc(Cl)cc(NC(c2cnn(C)c2C(=O)O)=O)c1I CC1(C)CCC(CCNC(C23CC2CN(C(=O)CN2CC4CC4C2)C3)=O)O1 N1(C(CC2C(CC)C2)=O)CC2CC(C1)N(C(c1ccc(Cl)c(C(F)(F)F)c1)=O)C2 C1(NC(c2cc(C)n(C)c2)=O)C2CC3C(C2)C13C(=O)NC1CCC(C)(C)C1 CC(C)(C(=O)NCC1CCCN1C(c1cn(CC(N)=O)nn1)=O)N1CCOCC1 Cc1cnc2cc(C(N3CC(=C(F)CNC(C4CCCS4)=O)C3)=O)ccn12 C(c1c(F)cccc1F)=CC(=O)NCC1C(C)CN(C(c2cccnc2)=O)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCC(C)(CO)NC(=O)CC2CCCN2C)c1Cl N1(C(c2ccc(CNC(C)=O)o2)=O)CC(C)CN(C(=O)Cn2ccnn2)CC1C c1(C(=O)NCCC2(C)CCN(C(C(CSC)C)=O)C2)ncc(F)cc1F N1(C(C(F)=CCC)=O)CCN(C(=O)CSC(C)C)C(C2CC2)C1 C1(OC(c2c(C)nn(C3COC3)c2)=O)CCN(C(=O)NCC2CCC2)CC1(C)C C1(NC(c2cnc(C)s2)=O)CC2CC(NC(c3cc4n(n3)CCOC4)=O)CC2C1 N1(C(Cc2n(C)c(S)nn2)=O)CCCC(O)(CNC(C2CC(C3CC3)=NO2)=O)C1 C(=O)(CCCCC(C)(C)C)N1CC(C(C(N2CCC(C#C)(O)C2)=O)O)C1 C1(C(N2CC(NC(c3c(OC)cccc3)=O)C(C)C2)=O)CCC(F)(F)CO1 c1(N(C)C)cc(Cn2cc(-c3cnc(-c4ccccc4)nc3)nn2)cn1C c1(C(=O)NC)ccc(C(F)F)cn1.c12csc(c1)CN(CC)CCNC2=O Nc1cc2c(cc1C(=O)NC(CNC(C1CC3CCC1CC3)=O)C1CC1)OCO2 N1(c2n(C3CCn4c(C)ncc4C3)nnn2)CCC2(CC1)CN(C)C(=O)O2 C(C1CCCc2ccccc21)NC(c1c(C)sc(Br)n1)c1nnnn1CC1CC1 N1(C2CCN(C(C(C)N(C)C)=O)C2)CCC(NC(c2ccn(C(F)F)n2)=O)CC1 CC(C)CCC(C)N(C)C(C1(CC)CN(C(c2cccc(O)n2)=O)C1)=O c1(C(=O)NCC(CC=C)NC(C23COC(CF)(C2)C3)=O)ncccc1CO N1(C(CSCC)=O)CCC(NC(=O)C(Cc2ccccc2)c2ccccc2)C1C N1(C(C(c2c(C)noc2C)CC)=O)CCN(C(c2ncoc2C)=O)C(C)C1 C(=O)(C(C)(C)C(C)NC(C1CC(CF)C1)=O)NC(C)Cc1ccccc1 Nc1cc(Cl)cc(Cl)c1C(=O)NC(C1CCCCC1)CNC(=O)C1CC1 N1(C(c2c(C(C)(C)C)con2)=O)CC2(CNC(C3(S(C)(=O)=O)CC3)=O)CCC1C2 Cc1cc(C#N)cnc1C(=O)NCCC(O)CNC(C1CCC(C)(C)CC1)=O CON(CCC(=O)NC1CC(C)CCC1O)C(=O)c1ccc(OC)cn1 CC(O)C(C)CNC(=O)C(C1CC1)N(C)C(c1ccn(CCF)n1)=O Cc1csc(C(N2CC3CC2(CNC(c2cnn(C)c2)=O)C3)=O)c1Br CC1(C)COCC(CC(=O)NC2CC3(C2)CC(NC(c2cnccn2)=O)C3)O1 C1(C)(C(N(CCCCN(C)C(C2CC(C)(C)C2C(F)(F)F)=O)C)=O)CNC(=O)C1 C1(NC(CC2CCCC(C)C2)=O)CN(C(c2coc3c2COC3)=O)CC1N=[N+]=[N-] c1(NC(c2c(C)oc(CNC(C3OCCC3C)=O)n2)=O)cnc2ccccc2c1 C1(CCC(=O)NC2CC(CCOC)C2)CCCN(C(=O)Cc2ccc[nH]2)C1 c1(C(N2CCC(CNC(COc3cc(C)on3)=O)C2)=O)nccnc1C(N)=O N1(C(C2(C)C(C)(C)C2)=O)CCC(CNC(c2ccc(Cl)o2)=O)C(O)C1 N1(Cc2c(-c3ccc(OC)cc3C)scc2)CCc2cccnc21 c1(C2(C(N3CCC(N(C(c4cc(C)ncc4)=O)C)C3)=O)CC2)ccnc(Cl)c1F C12(CNC(C(c3cncn3C)N(C)C)=O)CC(NC(=O)CC3(C)CC3(F)Cl)(CO1)C2 c1(C(N(C)CC2(O)CN(C(C(C(C)O)(F)F)=O)C2)=O)cnn2c1NCCC2 CC1=NOC(C)(C(=O)NC2CN(C(c3c[nH]nc3C3CCC3)=O)CC2O)C1 C(CN=c1nc[nH]c2c(C)cccc12)N(C(Cc1c(C)n[nH]c1C)=O)C N1(C(=O)OC(C)(C)C)CCC2(CC1)CN(C(c1nnn(C(C)(C)C)n1)=O)CC(C)O2 Cc1c(C(N2CC(NC(c3cccc(N)c3N)=O)CC2C)=O)cncc1Cl c1(C(=O)NCC2(CCCNC(C3(CSCC)CC3)=O)CCC2)cc(C)no1 C(C(=O)NOC(C)(C)C)(c1cccnc1)NC(C(C)N(C(C)=O)C)=O C(C(CO)(CO)NC(=O)C(O)CNC=O)N(C(C#CC=O)=O)C.N(C)C N1(C(C2(OCC)CC2)=O)CCN(CC)CC1.N1CC(C(C(=O)NC)OCC)C1 C1(N(C(C=CC=CCC)=O)CC)CCN(C(=O)C(c2ccccc2)C2CC2)CC1 c1(CNCc2c(OC)cc(OC(F)(F)F)cc2)cccn2ccnc12 C1(NC(C2CC(Cl)(Cl)C2)=O)C2CCN(C(c3cc(CO)[nH]n3)=O)C12 CC(C)C(C)(CNC(=O)COC(F)(F)F)NC(c1ncncc1F)=O N1(C(C(C)NS(CC)(=O)=O)=O)CCC(CNC(=O)CN(C)C)(OC)C1 C1(OC)CN(C(c2cc(C(F)F)nn2C)=O)CC1NC(=O)CCCF N1(C(c2c(CC)nc[nH]2)=O)CC=C(CCNC(C2C3C4CCC(C4)C23)=O)CC1 Fc1ccc(N2CCN(c3cccc(Br)c3)CC2)c(F)c1F c1(CSCC)ccc(C(N2CC(OCCNC(=O)CC3(C)CC3(F)F)C2)=O)cc1 C(C(C)CS(N)(=O)=O)SC.C1(C)(c2nnnn2-c2ccccc2)CCN1 N1(C(C(F)=CCC)=O)CCCC1C=CC(=O)NOCCC(C)C CCCS(=O)(=O)CC(=O)N1CCOCC(NC(C2CC(=O)N(C)C(=O)N2)=O)C1 C1(C(=O)NCC(CCCC)NC(C23CC4CC2C3C4)=O)CC(C(C)(C)C)=NO1 C1(CNC(c2cnc(OC)s2)=O)CC(C)N(C(c2snnc2C)=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NC2C3CN(C(=O)CC4CCC(=O)NC4)CC23)n1 c1(C2C(C)C2)nocc1C(=O)NC1(CCCNC(c2sccc2F)=O)CC1 CN1CCCC1C(N1CC(CCCCNC(C2(Cc3cccnc3)CC2)=O)C1)=O c1(C(=O)NC2(CCNC(C3(C)CC3)=O)CC2)cc(C(F)(F)F)ncc1Cl C(C)(CO)(C(=O)NC1CC1(C)C(F)F)NC(CC1(OCC)CC1)=O C1(CNC(C2(CC#C)CCCO2)=O)CCN(C(c2cnc(O)n2C)=O)CC1C CC1CN(C(c2csc(-c3ccoc3)n2)=O)CCC1CNC(C1(C2CC2)CC1)=O c1(C(=O)NCC(CNC(C2(C)COC2)=O)F)ccc2[nH]c(=N)[nH]c2c1 C(=O)(C(O)CCCNC(C1CN2CCC1C2)=O)NCc1cnc(COC)[nH]1 c1(C(=O)NC2CCCC(CNC(c3c(CC)occ3)=O)C2)cc2ncccc2[nH]1 c1(N2CCN(C(=O)OC(C)(C)C)CC2)ncnc2c1nnn2C1CC1.C1CCCN1 Cc1cc(C(N2CCC(CCNC(C3CCCS3)=O)C2)=O)ncc1Cl N1(C(Cc2scc(C)n2)=O)CCC(NC(=O)CCCNC(=O)C(C)(C)C)C(F)C1 C1(CC(=O)NCC2C=CC(NC(C3OCC(C)(C)C3)=O)C2)CCCC2(CC2)C1 O=C1Cc2c(C(N3CC(NC(=O)Cc4cncs4)C4(CCC4)C3)=O)cccc2N1 c1(-n2c(CCF)nc(C(C)SCC)n2)cc(Br)cn(C(C)C)c1=O S(=O)(=O)(c1ccc(N2CC3CC3C2)c(Br)c1)NC(c1cccnc1)CSC C1(NC(CC(c2ccc(Br)cc2)C)=O)CCC2(CC1)CN(C(C1CC1F)=O)C2 c1(SCC(=O)NC(CCOC)CNC(C2CCOC2C)=O)ccc(Cl)cc1 C1(CC(=O)NC2(CN(C(c3c(C)nc(C)[nH]3)=O)C)CC2)SC2=NCCN2C1=O c1(NC(=O)OC)cc(SN2CCOCC2C)ccc1[N+](=O)[O-].c12ccc(cc1)NC2 N1(C(c2cc(OCC)n[nH]2)=O)CCCC12CCCN(C(=O)C(O)CCC)C2 c1(CN(C(C2CCCCC2)C(=O)OC)CCCN(C)C)ccc2c(n1)CCCC2 c1(CC(=O)N(C(C)C(c2ccccc2)O)CC2CC(F)(F)C2)ccc2c(c1)CNC2 CCCCCCC(=O)N1CCC(C(C)NC(=O)CCc2ccon2)C1 c1(OC)ccc(Br)cc1C(=O)NC1(F)CCCN(C(c2ncn(C)n2)=O)C1 S(=O)(=O)(c1cccnc1N1CCC(CCCO)C1)NCC1(C)CCC12CCC2 C(=O)(C1=Cc2ccccc2C1)NC(CC(=O)Nc1c(C)noc1)C(C)(C)C CC1CN(C(c2cc(F)cc(F)c2O)=O)CC(C)C1NC(C1CCN(C)CC1)=O c1(CC(N2CC3CN(C(C4(C5CC5)CC4)=O)CC23)=O)c(Cl)cccc1Cl CCC(CC(=O)N1CC2COCC2(C(=O)NCCNC(=O)NCC)C1)C(F)F c1(N(C(c2ccsc2)C)C)ncnc2c1ncn2CC(O)C1CCC1 C(=O)(C1CNC(=O)c2ccccc21)NCC1CN(C(C=CSC)=O)CC12CC2 C=CC(O)C(=O)N1CC(F)(c2cn(CCC(=O)NC3(CS(N)(=O)=O)COC3)nn2)C1 C(=O)(CC1COc2cc(OC)ccc21)Nc1cc(C(=O)OC)c(OC)cc1 Nc1c(C(=O)NC2CCN(C(=O)C(F)(F)C3CC3)C2)cccc1[N+](=O)[O-] C1(CCNC(C(=O)NCC(F)F)=O)CCN(C(=O)CC2(N(C)C)CCCC2)CC1 c1(N2CCC(C)(C(N)=O)C2)ccc(Br)c(S(=O)(=O)N2CCC(N3CC(O)C3)C2)n1 c1(Sc2ccccc2)nccn1C(=O)NC1C(NC(c2cc(C3CC3)c[nH]2)=O)C1 N1(C(C(C)OC)=O)CCC2CN(C(c3cnn4ncccc34)=O)CC2CC1 C#Cc1cccc(CC(N2CCC(C)C2C(N2CCC2(C)C(=O)OC)=O)=O)c1 C1(CC(=O)NCC(CC)N(C(CC2N(CC)CCC2)=O)C)CCN(C)CC1 Cc1cc(Br)ccc1C(=O)NC1CC(NC(c2cc(F)ccc2O)=O)C1 C(=O)(CS(=O)CC)NCC(CC=C)NC(c1csc(C(C)(C)C)c1)=O c1(C(N2CCC(C)(NC(=O)Cc3ccccc3O)C2)=O)nnn2c1CSCC2 c1(C(N2CCC(CNC(c3c(C)scn3)=O)CC2)=O)nc(Br)cnc1N C1(C(N(C(CNC(C2(NC(=O)OC)CCCCC2)=O)C)C)=O)COC2(CCC2)C1 N1(C(CSCC(C)C)=O)CCCC(CNC(C2(n3ccnn3)CC2)=O)C1 C1(C(=O)OC)CC(=O)CC(=O)C1.C(C(O)CO)N(C(=O)C(C)N)C(C)C N1(c2[nH]c(=NCc3ccc(F)cc3F)cc(C)n2)CCN2CCN(C)C2C1 C(=O)(C(C(=O)N1CC2C(NC(c3cc(OC)cnn3)=O)C2C1)C(C)(C)C)NCC N1(C(c2ncn(CC)c2)=O)CC(CNC(c2cnnn2CC)=O)CC1(C)C C#Cc1cc(C(=O)NC2CCCCC2C(N2CCC(O)(CC#C)C2)=O)ccc1C N1(C(C2CCCN(C(CCCC)C)CC2)=O)CCCC(O)(CF)CCC1 C1(C(=O)NCCC(C)O)CCCCN(C(=O)C(F)CC2CCOC2)C1 CCC(CCCO)NC(=O)N(C)CC1CC1(F)F Cc1cc(OCC(C)SC2CCOC2)c(C)c(C)c1.C1CC(=O)O1 C(=O)(C(F)CC(C)(C)NC(=O)CC1(C)CCC1)N(C)CC1CCOC1 C(=Cn1nccc1-c1nc(-c2ccccc2)no1)OC c1(C(N2CC(C)C(NC(=O)COCc3ccccn3)C2)=O)c(O)ccc(Cl)c1O N1(C(Cc2c(C)noc2C)=O)CC(NC(=O)C(C)N(C)C)C2(CCC2)C1 N1(C(c2csnc2Cl)=O)CC2COCC2(C(N2CC3CCC2C(O)C3)=O)C1 CCC(O)C(=O)NC1CCCC1CNC(C1(NC(=O)NC)CCCC1)=O C(=O)(C(F)CCC(C)(C)C)N(C1(C(N(C)Cc2cccc(C)c2)=O)CC1)C C1(CCNC(CCC#N)=O)CN(C(c2ccc(-c3ncon3)cc2)=O)CCO1 N1(C(CCCC(C)=O)=O)CCC2(CCN(C(c3c(C)cccc3F)=O)C2)C1 c1(C(N2C(C)CC(NC(C(CC(=C)C)NC(C)=O)=O)C2)=O)cnc2ccccn12 CCCC(C(=O)N1CCC(C(F)F)(CNC(c2ncsc2C(F)(F)F)=O)C1)OC C=CCCCCCC(=O)N1CCCC(N(C(C2CC2(C)C(C)C)=O)CC)C1 c1(C(=O)OCC)ccc(F)c(NC(C2CC23CC(NC(=O)C(Cl)(Cl)Cl)C3)=O)c1 c1(OC)ncnc(C(=O)NC2(C)CN(C(C3CCOC3=O)=O)C2)c1F C1(C)(C(=O)NC2C(CNC(CC3(COC)CCCC3)=O)C2)CCCNS1(=O)=O c1(N(C2CCN(C(Cn3c(CCC)nnc3S)=O)C2)C)nc2cccc(F)c2o1 N1(C(=O)COCC2CCOC2)CCC(CNC(c2cnc(C(F)(F)F)s2)=O)CC1 C1(CNC(C(C)Cc2cnc[nH]2)=O)CC2(CCC2)CN1C(c1c[nH][nH]c1=N)=O C(C(C(=O)N(CC(C(=O)NC)n1cc(C(C)(C)N(C)C)nn1)C)N(C)C)OC n1(CCNC(C(Cc2ccoc2)NC(c2c(CC)n[nH]c2)=O)=O)ccccc1=O C1(C(=O)NC2(C)CCN(C(c3c(C(C)C)scn3)=O)CC2)CC2(C1)CC21CCC1 c1(C(N(CC(=O)OC)CC(=O)NC2CCC2SCO)=O)ccccc1.C(C)(C)(C)O CC1CN(C(c2nc(O)[nH]c(=O)n2)=O)CCN1C(=O)CCC1CC1(C)C c1(COC)nn[nH]c1C(=O)NCCCNC(C1(N2CCCC2)CC1)=O C(CCCC(C)(C)C)NC(CCOCCNC(C(COC(C)=O)(C)C)=O)=O C1(CCNC(Cc2c(C)n[nH]c2C)=O)C(C)CCCN1C(c1csc(CO)n1)=O C1(CCC)(C(=O)OC)CCN(C(=O)COCCNC(=O)CC2CC(C)(C)CO2)C1 c1(OC)cc(Cl)c(C(=O)NC2CC(NC(c3nnc(O)cc3O)=O)C2)cc1OC CCC(F)(F)CC(=O)N1CC2CC2C1C(=O)NCC1CSCCO1 C1(n2cc(C(C)OC)nn2)CC2CCC1(NC(=O)Cc1cncn1CC(C)C)C2 C1(NC(CCC(C)SC)=O)CCN(C(=O)CC(C)(C)C#N)C12CCC2 C1(NC(c2n[nH]c(CC)c2Cl)=O)CN(C(=O)C(C)NC(C)=O)CC12CCOCC2 NNCC.C(=O)N CC(C)(C)CCC(C)(c1nnnn1C1CC1)NCc1ncc(Br)s1 c1(C(N2CC(NC(c3ccc(CCC)[nH]3)=O)C(C)C2)=O)nc(O)[nH]c(=O)n1 C1(C(=O)NC2CC23CC(OC)C3)(CC)CCCN1C(=O)COCCCF CC1C(NC(=O)COC2CCC2)CCCN1C(c1ncoc1C(F)(F)F)=O Nc1cc(C(=O)NCC=CCNC(c2coc3c2CSC3)=O)cc(O)c1 C#CCCC(O)C(=O)NCCCCCN1CCN(C(=O)C(C)(C)C2CC2)CC1 CC(C)C(CCC(=O)NCCC1CC(F)C1)NC(C12CCC(CC1)CO2)=O C1(C(=O)NC2CCOC(C)(C)C2)(OC)CCN(C(=O)CCCCCSC)CC1 C12C3CC4CN(C1C4C3)C2=O.Cc1nc(C(C)NC(C)(C)C)oc1C c1(N2CC(c3c(CNC(c4c(C)con4)=O)nco3)C2)ncc([N+](=O)[O-])cc1Br C1(C(C(=O)N(CC(C)(C)NC(CSCC(C)C)=O)C)O)CCCCCC1 C(=O)(CCCC(=O)N(C)C)NC(C1CCN(Cc2ccc(C(N)=O)s2)C1)C c1(C(N(CCOCCNC(c2cc(C)ns2)=O)C)=O)cccnc1-n1nccn1 c1(C(=O)NC(CCNC(c2c(C)con2)=O)C)c(S(N)(=O)=O)ncn1C C(=O)(CCCCCCSC)NC1CC(C(C)NC(C(CCSC)O)=O)C1 N1(C(c2c(C)cns2)=O)C2CC1CN(C(C1(C)CCCCC1C)=O)C2 C1(C)(CNC(N(CC)Cc2cccc(Cl)c2F)=O)CS(=O)(=O)CCO1 CCC(CC(F)(F)F)C(=O)NCC12CC1CN(C(c1cc3n(n1)CCO3)=O)C2 C(=O)(C(O)P(C)(C)=O)NCC(CC(C)C)NC(c1c(C)ccn1C)=O CCC(CSC)N=c1cc(NCCC(=O)NC(C)C)nc(C(F)(F)F)[nH]1 c1(C(N2CCC(CCN(C(C(CC)N(CC)CC)=O)CC)C2)=O)cncc(C)c1 C(CS(=O)(=O)CC(=O)Nc1cccnc1C(=O)NC1(CO)CC2CCCC12)OCC c1(C(=O)NCCOCCN(C)C(C2SC3C=CC2CC3)=O)nc2ccccc2[nH]1 CCC(C(=O)NCCC1CC(NC(=O)CCCOCCOC)C1)OC C1(CN(C(=O)C(C)(C)F)CC)CCN(C(c2c[nH]nc2-c2ccncc2)=O)CC1 C(CCC(O)CO)NC(C1(CNC(C2CC(C(N)=O)C2)=O)CC2(CC2)C1)=O NS(=O)(=O)C1CN(C(=O)C(C2CCCCO2)F)C1 CC(C(=O)OC(C)(C)C)C(=O)N1CC(F)CC1CNC(=O)C=CC(N)=O c1(OCC(=O)NCC2N(C)CCN(C(=O)CNC=O)C2)c(F)c(F)cc(F)c1F c1(C(=O)NCC(C)NC(c2c(C)cncc2F)=O)cc(S(N)(=O)=O)co1 C1(NC(C=CCNC(c2ncc(OC)nc2)=O)=O)CCCCNC1=O CN=c1[nH]nc(CC(=O)NC2CCC2NC(c2csc(C)c2C)=O)s1 C1(CCC)CCC(C(=O)NC(C)=O)CC1.C12CCC(C1)N(C)CCCNC2=O c1(C(=O)CNC(=O)NC2CCCCC2)ccc(Br)cn1 C1(C2CCN(C(=O)Cn3ncnn3)C2)(NC(CC(C)(O)C2CCCCC2)=O)CC1 c1(C(N2C(CN(C(C(C=C)O)=O)C)CCC2)=O)cc(C)n(-c2ccccc2Cl)n1 CC(C)S(=O)(=O)C(C)C(=O)NC12CCC(CN=c3[nH]cncc3Cl)(OC1)C2 CCC(C)(F)C(=O)NC(CNC(=O)COCc1cccc(C)c1)C1CC1 Cc1c[nH]c(CC(N)=O)c1C(=O)NCC1CC(F)CN1C(C1CSCCS1)=O c1(NC(C2CCC(CNC(CSCCC)=O)CC2)=O)cc(C)ccc1F C1(NC(C2C(C)C2C)=O)CCC(CN(C(=O)Cc2ccc(CC#N)cc2)C)CC1 c1(C(=O)NCC2C3CN(C(C(CCSC)O)=O)CC32)cc(C)c(C)c(C)c1 N1(C(C(C2CC2)OCC)=O)CCCC1(CNC(C1(Cl)CC1)=O)COC N1(C(c2ccc(OC)o2)=O)Cc2ccc(CNC(=O)C#CC3CCOC3)cc2C1 c1(C(=O)OC)cccc(-c2ccc(NS(=O)(=O)CCC3CCOC3)cc2)c1 C(=O)(C1=NNC(=O)CC1)N1C2CC(NCc3c(C)nccc3)C(C2)C1 c1(C(N2CC3(C2)CN(C(C2CN4CCC2CC4)=O)C3)=O)ccc2nc(S)oc2c1 C1(CNC(CC=C=C)=O)CCN(C(c2c(C)nn3ncccc23)=O)CC1C1CC1 C1(NC(c2nocc2Cl)=O)CN(C(C2C=CCCC2)=O)CC1C(F)F C1(CNC(C(=O)NCCNC(C)=O)=O)CC2CCC1N2C(C1(CO)CC1)=O c1(C(=O)NCCCNC(CN(c2ccc(Cl)cn2)C)=O)cc2sccc2s1 C12(COC)CN(C1)C(=O)C1CCC1C2.C1(COCC(=O)N)CCCCC1.C(N)(=O)N CCC(CCc1ccccc1)C(=O)NC1CCN(C(C2CC(OC)C2)=O)C1 Cc1cc(=NCCC(C)NC(c2cnn(C)c2N)=O)c(C#N)c[nH]1 c1(NC(C(N2CCN(CC(C)C(=O)NC=O)CC2)C)=O)cc(S(C)(=O)=O)ccc1F C1(CCC)CN(C(c2c[nH]c(=NC)s2)=O)CC1NC(c1ccc(C(N)=O)cn1)=O c1(NC(C(=O)NCCSCC#C)=O)ccc(C(C)O)cc1 C12(NC(C(=O)NCC)=O)CC1CN(C(C1(C)CCNC1=O)=O)C2 C1(CNC(CC(C=C)c2ccccc2)=O)CC2(CO1)CN(C(C1CCCS1)=O)C2 c1(CC(C(=O)NC(C)CNC(=O)Cc2cncn2C)C)ccc(F)cc1F C1(C(F)(F)F)CCCC(NC(=NCc2ccnc(C3CC3)c2)NC2CC=CC2)C1 N1(C(c2cnc(S)nc2)=O)CCCC2(CCCN2C(=O)COC2CC(F)(F)C2)C1 N1(C(c2cc(OC)no2)=O)CCC(CNC(C2CCCCN2N=O)=O)C12CCC2 C(=O)(C(CNC(c1ccccc1C)=O)C(C)C)NCc1onc(C)n1 n1(CCNC(c2ccc(F)c3cnccc23)=O)cnc2cc(F)c(F)cc12 c1(N2CCC(C#N)C2)nccc(=NCCOC(=N)O)[nH]1.C1CCO1 N1(C(COC(CC)C)=O)CCCC2(C1)CN(C(c1cc(Cl)c(F)cc1Cl)=O)C2 Cc1cnc(O)c(CNC(C2(NC(C3C=CC=CC=C3)=O)CCSC2)=O)c1 c1(C(=O)NCC2C(NC(C(C)CC3CC3)=O)C2)ccc2c(n1)OCC(=O)N2 c1(CNC(=O)Nc2cc(C(F)(F)F)ncc2-c2ccnnc2)c(Cl)cccc1Cl Cc1sc(C(N2CCC(C)N(C(C3CCS(=O)(=O)C3)=O)CC2)=O)cc1[N+](=O)[O-] N#Cc1ccc(F)cc1CN1CC(NS(=O)(=O)c2cn[nH]c2)C(F)(F)C1 N1(C(C2(C)CN(C(CC3ON=C(C)C3)=O)C2)=O)CCN(C)CC1CCO c1(CCC)cc(C(N2CCC(CN(C)C(C3CC(OC(F)F)C3)=O)C2)=O)nn1C N1(C(C#CC(C)(C)O)=O)CCC2(CCC(CNC(=O)CC3CC4(CC4)C3)O2)CC1 CCCCC(C)(F)C(=O)NCC1COCCN(C(=O)C(C)(C)O)C1 N1(C(CC2(C)CC2)=O)CC(C2(NC(c3ccc(O)nn3)=O)CC2)C1 N1(C(=O)NCC(C2CCC(C)(C)C2)(C)C)Cc2ccc([N+](=O)[O-])cc2C1 O=C1Nc2cc(C(=O)NCC(CO)NC(=O)C=C(Cl)Cl)ccc2C1=O S(=O)(=O)(c1ccc(Br)c([N+](=O)[O-])c1)N1CC2CN(C(=O)C(CO)c3cccs3)CC21 C12(C(=O)NCCC(C)NC(C3CC(F)(F)C3)=O)COC(CS(C)(=O)=O)(C1)C2 N1(C(C(CC)c2ccccc2)=O)CCCN(C(c2c(C)n[nH]c2C)=O)C(CO)C1 c1(CCNC(c2snc(OC)c2Br)c2nnnn2CCCF)cccc(Cl)c1F C1(C(C(=O)Nc2c(C)nsc2)C)CCN(C(c2ccnn2C2CC2)=O)CC1 c1(NC(C)=O)ncc(C(N2CCCC2C(C)NC(C2CN(C(C)C)C2)=O)=O)s1 C1(NC(c2cc(Br)c(CO)o2)=O)CC2(C1)C(C(=O)O)C2(F)F C1(NC(Cc2nc(C)[nH]n2)=O)CC2CC1N(C(c1nc(C(C)(F)F)cs1)=O)C2 CCCC(C(=O)NC(C)CC1CCC1)NC(=O)CC1(N(C)C)CCC1 C(=O)(C(CNC(=O)CCOCC(C)C)CC)N(CCC)CC C(N=c1cc(C(C)(C)C)nc(Cl)[nH]1)C1CC(NC(CN(C)CC)=O)C1 C1(C(=O)OC)CCC(C(=O)NCC(C2CC2)NC(C2CCC(C(N)=O)C2)=O)CC1 c1(C(N(C(=O)Cc2c[nH]nc2C)CCC)C)nnc(COC(C)(C)C)n1C C(c1c(Cl)cccc1Cl)=CC(=O)NCC1CC(NC(C2CCCC2(F)F)=O)C1 n1(CC(=O)N(C(C)C(=O)NC(c2noc(C)n2)C)CC)ncccc1=O c1(C(=O)OCc2cccc(NC(CC)=O)c2)nc2ccccn2n1 CC1=CCCN(C(=O)CCC2(NC(=O)C=C3CCCCC3)CCCC2)C1 C(CC(C)(C)C)(C(=O)NC(CC(N)=O)C(=O)NCC(C)Cn1cccn1)OC c1(CC)nn(C)c(CC)c1S(=O)(=O)N1CCC(O)(c2nc(C(C)C)no2)C1 c1(C(N)=O)c[nH]c2ccccc12.C1(N(C(CN)=O)CC2CC2)C2CCC1CNC2 C1(C(=O)NC2CCC(NC(C3(CC#C)CCCCC3)=O)CC2)CNC(=O)CC1C c1(C(N2CC(CNC(CC(=O)NCC#C)=O)C(C)CC2)=O)cccc2oncc12 C(CCCCCC(=O)NC(c1n[nH]c(C)n1)C)NC(C1(CC)CCCO1)=O c1(OCC(=O)NC(C2CCN2C(=O)CCc2cc(C)no2)C)ccc(CO)cc1 c1(C(=O)NC2CCN(C(c3c[nH]c(=NC)o3)=O)C2)c(C)ccc(C)c1C Cc1nc(C(C)(C)C)ncc1C(=O)NC(CO)C(C)NC(=O)CC1C=CCCC1 C#CC(C(=O)NOCC(N1CCN(CC2CCC2)CC1)=O)C(C)C N1(C(C(C)(CO)NC(C(C2CCC(=O)N2)C)=O)=O)CC[Si](C)(C)CC1 c1(C(=O)NCC2(NC(C(C)=CC)=O)CCCCC2C)c(F)c(F)c(F)c(F)c1F c1(OC)cc(C(=O)NCC(C)NC(c2nc(C)n(C(C)C)c2C)=O)cc(F)c1 CC1CN(C(=O)C2=COCCO2)CC(C)C1NC(C1Cc2ccccc2O1)=O C(C(C)C(=O)OC)NC(C1CC(C(N(CCOC)C2CC2)=O)C1)=O c1(NC(C2CCCN(Cc3ccc(OC)nc3)C2)=O)ccnc(Br)c1F C(=O)(C(C)(C)CN(C)C(C1CC(C)N(C)C1)=O)NCC(C)OC1CCCCC1 C1(C(=O)NCCNC(c2cnc(CC(C)C)[nH]2)=O)COc2ccc(O)cc2O1 c1(CC(N2CCC(C#N)(c3cccc(F)c3)C2)=O)ccc2c(c1)CCCC2 c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)CCc3nnc(CN(C)C)o3)C2)c1 CCCCC(F)C(=O)NC(CC(=O)NC1C(O)C2CCOC12)C(C)C CS(=O)(=O)CC(=O)NC1C2CN(Cc3ccccc3)CC12.C12CCN(CC1)C2=O c1(C(N2C3C(NC(C4C(C=C)CC4)=O)C(C3)C2)=O)cc2ccc(Cl)cc2o1 CP(C)(=O)CCC(=O)NCC(CNC(=O)C(c1cccc(F)c1)O)CO N1(C(C)=O)CC2(CCN(Cc3ccc4c(c3)OCO4)CC2)CC1C(=O)O C12(CCC)N=C3N=C(NS3)CN(CC1)CC2.C1(CC(=O)OC)CCCOCC1 N1(C(C(C)NC(N)=O)=O)CC2(NC(=O)CC3(C)OCCO3)CCC1C2 CCCC(CNC(=O)CCc1cncs1)C(=O)NC1CN(C)CC1(F)F N1(C(C=CC)=O)CC(OC)C(NC(=O)COc2cccc(-n3cnnc3)c2)C1 C=CCC(F)(F)CNC(=O)C(C1CCN(C(C2CC23CC3)=O)C1)C Cc1ccc(C(C)C)cc1C(=O)NCC1CCCN1C(C1SC2C=CC1CC2)=O N1(C(CCc2cncc(C)c2)=O)CC(NC(=O)C=CCF)C(C)(C)C1 Cc1cc(CCC(=O)NCC(C)NC(c2c(C)nsc2Br)=O)cc(C)c1 Cc1cc(C(N2CCCC2C(C)NC(=O)CC(O)c2ccccc2)=O)nn1C CCC(CC)(CC)C(=O)N1CCC(C2(NC(c3ccn(C(C)C)n3)=O)CC2)C1 c1(C(=O)NCC(CNC(Cn2nc(C)n(CC)c2=O)=O)F)cc2ncccc2[nH]1 CS(=O)(=O)C1CCN(C(C2CN(NCc3nc(C4CC4)cs3)CCC2O)=O)C1 Cc1ccc(Cl)cc1OCC(N1CCCC(C(C)NC(c2cccn2C)=O)C1)=O CCC(CC(=O)NCC(C(=O)NCCN1CCC(CSC)C1)OC)C(C)C C1(NC(Cc2cnc(C)s2)=O)CC(C(=O)N(C2CC2C2CC2)C)C1(C)C O=C1Cc2cc(NC(c3ccc(-c4ccc(O)cc4CO)nn3)=O)ccc2N1 CCC(CCCC(=O)NCC(c1ccsc1)O)NC(=O)C(F)C(CC)CC C(=O)(C1=NOC(CNC(c2sccc2Cl)=O)C1)NC(CC)(C)C1CC1 Cc1ccc(C(N2CC3(CC3)CC2CNC(C2CSCCS2)=O)=O)cc1N c1(OC)cc(C(N2CCC(CC(N3CCCCC(C)C3)=O)C2)=O)cc([N+](=O)[O-])c1 C12(NC(COCCC)=O)CCOCC1CN(C(=O)CSC1CCC1)C2 N1(C(c2ncc(CC)cn2)=O)CCC2C(CCCN2C(C2COCCO2)=O)C1 CC1=C(C(=O)NC2CCCN(C(c3cc(C(F)(F)F)nn3C)=O)C2)CCC1 c1(C(N2CC(NC(CC#N)=O)C(CC3CC3)C2)=O)ccc2nncn2c1 CCC(C(=O)N1C(C)C2CC1C2NC(=O)COc1cnn(C)c1)C(F)(F)F c1(OC)ccc(CNC(C)=O)c(OC(=O)C(c2ocnc2C)N(C)C2CC2)c1 CC(C)CC(C(=O)NC1COCCC1NC(=O)Cc1nc(C2CC2)cs1)C(C)C Cc1nccc(-c2cn(C3CCN(C(=O)Cn4ccnc4C(C)C)CC3)nn2)n1 CCCC(C(O)C(=O)Nc1cncc(F)c1)NC(=O)CC(F)(F)C(F)F C=CC1(C(=O)NCC2(COC)CN(C(C3CC(C#N)(OC)C3)=O)C2)CCOCC1 c1(NC(C)CC(C)NC(c2ccc(C(C)(C)C)nc2)=O)nc(C#N)c(Cl)s1 c1(C(N2CCCCC(CNC(C3(CC(C)C)CC3)=O)C2)=O)ccc2occc2n1 CCCC(CC)C(C(=O)NCc1ncccc1OC(C)=O)N1CCS(=O)CC1C C(C1CN(C(C2CCC(=O)O2)=O)Cc2ccccc21)NC(CCC=C(C)C)=O Cc1c(CC(=O)NC(C2CN(C(C3C4CCCC34)=O)C2)C)cccc1[N+](=O)[O-] N1(C(C(C2CC(F)(F)C2)OC)=O)CCC(C(=O)NCCC(=O)OC)C(C)C1 c1(N2CCC(F)(CNC(c3ccc(F)nc3)=O)CC2)c(F)cccc1[N+](=O)[O-] CN1CCC(CNC(C2CNCCN2Cc2ccnc(Br)c2)=O)CC1 N1(C(CS(C)(=O)=O)=O)CC(NC(c2ccc3nn[nH]c3c2)=O)CC12CCOC2 c1(CNC(CCN(C)CCO)=O)cn(CCNC(=O)CSCC(F)(F)F)nn1 C1(NC(C(=O)NC)(C)C)CCN(CCNC(C2CC23CC3(F)F)=O)CC1 c1(-c2cn(CCC(=O)OC)nn2)ccc2cnccc2c1.C12CN(CC1C)C2=O Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(C2COCCO2)=O)CCC(O)C1)=O CC(C(=O)NCC(C1CC1)N(C)C(c1cn(C2CCOC2)nn1)=O)C(F)(F)F c1c(C)ncnc1C.C1(OC)CC(CNC(=O)OC(C)(C)C)N(C(=O)C2CC2)C1 N1(C(C(CC(=O)OC)C)=O)CC2CC1CCC2NC(c1ccc(C2CC2)s1)=O Cc1ccc(Br)cc1C(=O)CCC(=O)N(CCS(C)(=O)=O)C N1(C(C(C)CC(N)=O)=O)CCCCC12CN(C(=O)C(C)(C)CO)C2 c1(C(=O)NCC2OCCN(C(c3cnc(OC)s3)=O)C2)ccc(Cl)c(F)c1N Cc1nnccc1C(=O)NCC1CN(C(=O)Cn2ccccc2=O)CC1C C1(NC(=O)C=Cc2cocn2)C2CCC1N(C(C1(C3CCCO3)CCCC1)=O)C2 CCS(=O)(=O)CCNC(=O)C(n1cc(CO)nn1)Nc1ccc(C(C)=O)cc1 c12cccc(c1)CCC(=O)NC2.C(N=c1[nH]ncs1)C1(C)CC1c1ccccc1 Cc1ccc(C)c(C(N2CC(O)(CO)C2)=O)c1.C12CC(C1)CCNC(=O)C2 C(=O)(C(F)CC1CC1)N(C1(CNC(=O)C(O)(C2CC2)C2CC2)CC1)C c1(C2(C(N3CC(n4cc(C(CSCC)(C)O)nn4)C3)=O)CC2)c(F)cccc1Br c1(SCCN(C(c2ccnc(NC)c2)=O)NC(COCC)=O)ccc(F)cc1Cl N1(C(c2cccc(O)n2)=O)CC2OCCN(C(=O)CC(O)c3ccccc3)C2C1 N1(C(CC2CCCN(Cc3cc(Cl)cc(C(=O)O)n3)C2)=O)CCn2ncnc2C1 c1(C(N2CC3C(NC(C4(CC5CC5)CC4)=O)C3C2)=O)cnc2n1CCS2 C(c1cc(Cl)ccc1OC)=CC(=O)NCC1C(NC(CC2(OCC)CCC2)=O)C1 C1(C(=O)NC(CC=CC)C(=O)NCc2nc(C)cs2)CCCC(C#N)C1 C(=O)(C(C(C)(C)C)N(C)C)N1C(CN(C(CCN(C)CC)=O)C)CCCC1 C(=O)(C(O)CC(F)(F)F)N1CCCC(C)(c2ccccc2)C1.n12cc(nn1)CC2 C1(C(=O)NCCCC2N(C(C3CCC(C)C3)=O)CCC2)CC2CCC1O2 Cc1cn2cccc(C(=O)NC3C=CCN(C(c4cnn(C)n4)=O)C3)c2n1 N1(C(c2cc(CC(=O)OC)on2)C(=O)NCC(=C)C)CCCCC1C1CCCC1 N1(CC=C)C(=O)c2ccc(C(N3CCN(C(C4(C)CC4)=O)C(C)C3)=O)cc2C1=O Cc1nc(N2CC(CNC(=O)Cn3cc(C)ccc3=O)CC2C)cc(O)n1 C1(C(N(C)CC2(OC)CCC2)=O)CCCC(NC(=O)CCCc2ncco2)C1 CC1CN(C(c2c[nH]nc2F)=O)CCN1C(c1cc(F)ccc1O)=O c1(CC(OCC)OC)ccccc1C(C)NC(=O)NC12CCCCC1C2 CCC(CC)(CCOC)C(=O)NCCC1CC2CCC1CC2 C#CCC(C(=O)NCC1(C(C)O)CC1)NC(=O)CC1CC1CC c1(NC2CC(CC(C)C(=O)NC(=O)C3=CS(=O)CCC3)C2)ccc([N+](=O)[O-])cc1Cl N1(Cc2c(OC)cco2)C(C(=O)N(c2cc(C)ccc2C)C)CC2CCCCC12 c1(C(C(=O)NC2CCC(NC(c3c(C)cno3)=O)C2)C)ccc(Cl)cc1 N1(C(CCCSC)=O)CCCC(C2(NC(C3(C)CC3Br)=O)CC2)C1 c1(OC)ccc(N)c(C(=O)NCC2CC(NC(C3CC3(C)C(C)C)=O)C2)c1 c1(OC)cc(C(=O)N(CCCNC(C2(C)COCC2(F)F)=O)C2CC2)cc(F)c1 c1(C(N2CCC(NC(C(CC)C3CCOCC3)=O)C2)=O)ccc(O)cc1C c1(NC(CC(CC2CC2)NC(C2C(=C)C2)=O)=O)c(C)cc(O)cc1C C1(N(C(c2ccc(C(C)C)o2)=O)C)CN(C(C2CCCOC2)=O)CC12CC2 CC(C)(C(=O)NC1CC1CNC(=O)C(C)(O)C1CCC1)NC(=O)C(F)(F)F C12(C(N(CC(CNC(c3n(C(C)C)cnc3)=O)O)C)=O)CCOC1CC(=O)NC2 C=CCC(CC(C)C)C(=O)NC(CC(=O)N(CC#CC)C)C(F)(F)F c1(CC)nc(-c2cnc(Br)s2)n(C2(c3ccsc3)CC2)n1 C1(C)(NC(C2C(C)C2)=O)CCN(C(=O)CCCC2CC2)C1 CS(=O)CCC(=O)NCCC1CCN(C(=O)C=CS(C)=O)CC1 N1(C(c2c(OC)cc(F)cc2)C(=O)NC2COC2)CCN2C(=O)CCC2C1 c1(SC(C)C(N2CCC(CN(C(=O)COCC(F)(F)F)C)C2)=O)ccccc1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(NC(c2ccc3occc3c2O)=O)C1 C1(NC(COC(CC)(C)C)=O)CC1C1CCCN(C(=O)C(C)OCC(C)C)C1 Cc1nccc(C(N2CCC(C)CC2CNC(c2ccnn2C)=O)=O)c1O C1(NC(c2ccncc2)=O)CCC(NC(c2sccc2I)=O)CC1 CCC(C)(C(=O)N1CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C2(CCC2)C1)C(F)F C1(C(=O)NCC2CN(C)C2)CN(C(c2cc(Br)nc(Br)c2)=O)CC(F)(F)C1 CC1C(NC(=O)CC2CC(C)(C)CO2)CCCN1C(C1CC2(CSC2)C1)=O c1(NCc2c(Br)cc(C)s2)ccc(C(=O)O)c(C)c1C c1(C(=O)NCc2ccc(C(=O)NCC(CC)O)cc2)ccc(C)c(O)n1 C1(N(C(C(C2CC2)OC)=O)CC2CC2)CCN(C(C2CC3CC3C2)=O)CC1 CC(CC(O)c1cccs1)NC(=O)CCC1(C(F)(F)F)CC1 C(=O)(CC(C)C(=O)OC)NC(CSCC)C(=O)NCC(C)(O)CC N1(C(c2cc(CC)[nH]n2)=O)C2CCC1CN(C(c1[nH]c(C)c(C(C)=O)c1C)=O)C2 CC(C)CS(=O)(=O)CCC(=O)NC(CNC(c1ccccc1N(C)C)=O)C1CC1 c1(CNC(=O)NCCCCNC(=O)OC(C)(C)C)ncc2ccccc2n1 CC(CC(=O)N1CCCCC1CCC(=O)NCC(C)(O)CO)C(F)(F)F CC(C)CCCCC(=O)NC1CCCC(NC(=O)Cn2cc(C#N)cn2)CC1 c1(OC)nc(N2CC(O)(CNC(=O)CCc3nnc(C4CC4)o3)C2)nc(C)c1F Cn1cc(C(=O)NC2CC(C)(C(=O)NCCOC3CCCC3)C2)ccc1=O C(=O)(C1(C)COc2ccccc21)NCC1C(NC(C=Cc2cc(OC)ns2)=O)C1 C1(CC(=O)NC(C)(C)CCCO)CN(C(C2CCCN2C=O)=O)CC12CC2 c1(NC(C2CN(c3ncc(F)cn3)CCS2)=O)c(O)cccc1[N+](=O)[O-] C1(C(=O)NCCCC(C)NC(c2c(OC)nccc2)=O)CCCCCCC1 CC(C)CC(CNC(=O)CCc1cncnc1O)NC(=O)CO c1(C(N(CCNC(c2nc(C(COC)C)sc2)=O)C)=O)ccc2c(c1)CNC2=O C=C=CCCC(=O)NC(C)C(C(C)C)NC(c1cnc(NC)cn1)=O c1(CCC(=O)NC(CCNC(C(CC)C)=O)C)cc(C)nc(C)c1 C12(NC(c3ccccc3)=O)CC1CN(C(c1cncnc1)=O)C2.C1(=O)CCCN1 n1(CC)nc(C(=O)NCCOCC(=O)N(C(C)CN(C)C)C)cc1O N1(C(c2ccc(C)c(Cl)c2)=O)CCCN(C(=O)C(C)C2(O)CCC2)CCC1 C1(NC(C=CCC)=O)CCN(C(=O)CSc2ccc(C#N)cc2)C(C2CC2)C1 C123CCCN(CC1C2)C(=O)c1noc(C)c1C(=O)N3.C(C(=O)NCCOC)OC C1(NC(C(CC(C)C)O)=O)CN(C(=O)Cc2ccc(Cl)cc2Cl)CC2CCCC12 c1(OC)ccc(C(=O)NCCCCNC(=O)Cc2cocn2)c(F)c1Cl c1(C(N2CCC(C3CCC3)CC2)C(=O)NCC)ccc2c(c1)CCCC2 CC1CCCC1(O)CNC.c1(C(=O)N)cccc(C(=O)O)c1 C(=O)(C(F)C(F)(F)F)N1CCCC(C(N2CCC(OCC#C)CC2)=O)C1 N1(C(CC(CCCC)O)=O)CCC2(CC1)CN(C(=O)C(O)C(F)F)C2 c1(N2CCCC(C)(C(=O)NC3CC(C)(C(=O)OCC)C3)C2)ccccc1[N+](=O)[O-] C1(COC(c2c(-c3cn(C)nc3)c[nH]c2)=O)CCC(O)CN1C(=O)OC(C)(C)C CCC(CC)CC(=O)N1C2CC1CN(C(C1CC1C(=O)OCC)=O)C2 C(=O)(C1CCCc2ccccc21)NC1(CNC(=O)CC2(O)CCOCC2)CC1 C(CO)(CCCCNC(C1C2CC3C(C2)C13)=O)NC(C1(CC)COC1)=O c1(C(N2C(C(=O)NCc3ccc(O)cc3)CCC2)=O)cc(F)cnc1Cl CC1(NC(c2ccncn2)=O)CCCCC1C(=O)NCC1(CO)CCC1 N1(C(C=CC(CC)C)=O)CCC(CNC(c2cnc(OC)s2)=O)(COC)CC1 CC1C(=O)N(CC(=O)NCC2(NC(c3cnn[nH]3)=O)CC2)C(=O)C1C N1(C(c2c(C)n[nH]c2C)=O)CC2(NC(C3CCOC3C3CC3)=O)CCC1C2 N1(C(CCc2c(C)ncs2)=O)CCN(C)C(CNC(=O)Cc2cnoc2)C1 C1(C(=O)NCCC(=O)NCC(C)C)CSCCN1C(=O)Cc1cncnc1 C1(C(=O)NC23CC(CNC(C=CCCC)=O)(C2)C3)C(C(F)(F)F)C1[N+](=O)[O-] CCC(C(=O)NCCCNC(c1cccc2[nH]nc(O)c12)=O)C(C)(C)CC C1(F)(CNC(=O)CC2CCOC2)CCCN(C(=O)CCc2cnoc2)CC1 N1(C(CCC)=O)CCC(O)(C(=O)OCC(c2ccccc2)O)C1 Cc1ccc(F)c(C(=O)NC(C)CC2CN(C(c3ccc(OCF)cc3F)=O)C2)c1 C1(C(=O)Nc2ccc3oncc3c2)CCc2nc(-c3cncc(F)c3F)sc2C1 Cc1c(O)c(=O)ccn1CC(=O)NCC(CNC(=O)C(F)C(C)(C)O)C(F)(F)F N(C(=NCC(F)F)NCC(O)C1CCC1)C1CC(CC(C)C)C1 C=CCCCCCC(=O)N(CC(=O)NC(C1CCCO1)CO)CC1CC1 c1(CN(C(C(=O)NC(C(C)C)Cc2cccc(Cl)c2)=O)C)ccc(C(N)=O)cc1 c1(C(=O)NCC2(F)CCCN(C(C(C)(C)OC(C)=O)=O)C2)ccc2nn[nH]c2c1 c1(C(=O)NCC2C3CN(C(C4CC(=O)N(O)C4)=O)CC23)ccnc(O)c1 c1(NC2C3N(C(CC(C(C)C)O)=O)CC(CC3)C2)ncc2scc(C(F)F)c2n1 c1(C(=O)NCCN(C(C(=Cc2ccccc2)OC)=O)C2CC2)cc(O)cc(=O)o1 C(CN=C(NCC1(OC)CCOC1)NC1CC1c1ccc(C#N)cc1)SC C(CCCCC(=O)NCC(C)(C)C(=O)Nc1ccc(C(N)=O)cc1)=CC N1(C(C(c2ccc(C)s2)C)=O)CCN(C(=O)CC2CC3(CC3)C2)C(C)C1 c1(OCC(=C)C)ccccc1CN1CCCC(C(=O)NC(c2nnc(C)s2)C)C1 C1(CC)CCCCCC1(c1nnnn1C(C)(C)C)NCCc1cc(Cl)sc1Cl c1(CCC(=O)NCCN(C(C2(Cl)CC2)=O)CC)ccc(OC)cc1F C1(C(=O)NC(CNC(C2C(OC(C)=O)C2)=O)(C)C)C=C(C)CS1 C1(C(=O)OC)CCN(C(=O)NC2CC2c2ccccc2)CCO1.c1ccnn1CO N1(C(C2(CCCC)CC2)=O)CC2CC(NC(c3coc(Cl)n3)=O)C1C2 C1(CC)CN(C(c2cccnc2OCC)=O)CCC1NC(=O)C=Cc1cc[nH]c1 C1(CNC(CC2C=NN(C)C2=O)=O)CCCCN(C(=O)C=CC2(C)COC2)C1 CCCCC(CNC(=O)CC1(OC)CC1)NC(=O)CCc1ccon1 C(=O)(CC(CC(C)C)NC(c1scc(C)c1C)=O)NC(CC)Cn1cncn1 C(CN=c1[nH]cnc2ccc(F)cc12)(C1CCCC1)NC(c1ccc(Cl)o1)=O Cn1cc(C(=O)NCCC(C)(C)CNC(c2cnc(O)c(F)c2)=O)ncc1=O C1(NC(=O)CC2CC(F)(F)C2)CC(F)CN(C(=O)CCSCc2ccccc2)C1 n1(C(CC)C)nc(-c2cccc(C(C)OC)c2)nc1-c1n[nH]c(O)n1 C(=O)(C(C)(C)CS(C)(=O)=O)NC(C)CC(C)NC(c1cc[nH]c(=N)c1)=O c1(C(N2CCCC(CN(C(=O)C(F)C3CCC3)CC)C2)=O)ncn2ccccc12 Cc1nn(C)cc1C(=O)N(C(CNC(c1csc(C)c1N)=O)C1CC1)C Cn1cc(NC(C2CCC(F)(F)C2)=O)nc1C(=O)NC1CNC(=O)C1 c1(C(=O)NC(C2CN(C(C(C=C=C)C)=O)C2)C)coc2c1C(=O)NCCC2 CC1(CNC(=O)COCCCF)CCN(C(=O)CCc2cncs2)C1 N1(C(c2cccc(OC)c2)=O)CC2(C1)CN(Cc1ccc(OC)c(OC)c1)C2 CCCC(CC1CCCC1)C(=O)NC(CNC(C1(CF)COC1)=O)CCCC C#CCC(C(=O)NCCN1CCC(OC)C1)NC(=O)COCC(C)C C1(NC(=O)C=CC2CCC2)CCN(Cc2ccc(Cl)cn2)CC1F c1(C(=O)NCCN(C(=O)C(C(C)C)C(C)C)CC)cc(Br)c(C)cc1O c1(C(N2CCC(OC)(CNC(C3CCC3)=O)C2)=O)c(C)cc(C)c(Br)c1C c1(C(N2CC=CC(NC(C(C=C)(C)CC)=O)C2)=O)cnc(S(C)(=O)=O)n1C c1(CC(=O)N(CCC(C)NC(=O)CC2CCCN2C)C)ccc(F)c(Cl)c1 C1(NC(CNC(C)=O)=O)CC(CNC(c2cc(C(F)(F)F)on2)=O)C12CCC2 C(CN=c1[nH]c2ccccc2o1)N(CC)CC.n1(CC=O)cnnc1 C1(CNC(C(n2ncc(C)c2)C)=O)CC(C(=O)NCCO)=NO1.C1C(=O)N1 C=CC(CC)C(=O)NC1(COC)CN(C(C2(O)CCCC2)=O)C1 C(=O)(CC(C)c1ccco1)N(C(CNC(c1cnc(C2CCC2)[nH]1)=O)C1CC1)C C1(C(N2CCN(C(C3C(CCC)CCC3)=O)CC2)=O)CCC2CC1C2(C)C N1(C(CCN(CCC)C)=O)C2CCC(C2)C1CC(=O)NC1(O)CCC1 c1(C(=O)Nc2cccc(NC(C3N(C)CCOC3)=O)c2)c(N)cc(Cl)cc1F C(=O)(CCC(=O)NCCC(N)=O)NCC(CNC(C1(C)CCCCO1)=O)OC c1(C(=O)NCCCN(C(=O)CC2CCC(C)(C)CO2)CC)[nH]nc([N+](=O)[O-])c1Cl N1(C(C2C(C#C)C2)=O)CCOC2(C1)CN(C(=O)C(CC=C)CC(C)C)C2 Cc1nc2ncc(C(=O)NC3CCN(C(c4ccoc4)=O)CC3CO)c(=O)n2[nH]1 C#CCC(O)C(=O)NCCN(CC(C)O)C(c1cnc(-c2ccccc2)s1)=O N1(C(c2c(COC)ncs2)=O)CC(C)N(C(c2ccn(CC(C)C)n2)=O)CC1C CN1CCN(C(C2C(C)(C)C2(F)F)=O)CC1C(=O)NC1CN(C(N)=O)C1 c1(C(N(C(C)CNC(C2CC=CCC2)=O)CC)=O)csc(COC)c1 C(CC(C)C)(C(=O)NC1CCCCC1COC)NC(C(C(=O)OC)C)=O C(C)(CCC(=O)NCC(c1ccccc1)NC(C1(C)CC(=O)C1)=O)OC N1(C(CCCSC(C)(C)C)=O)CC(O)C(O)C1CNC(=O)CC=CC(C)(C)C c1(CC)cc(C(=O)NCC(CO)NC(=O)CNC(C2CCCCC2)=O)cn(C)c1=O CCCCS(=O)(=O)CC(=O)NC1(C)CCN(C(c2cc(C)c(C#N)cn2)=O)CC1 C(CCC(=O)NC(C1CCCC1)CNC(=O)C(C)NC(=O)COC)OCC C(=O)(CCC(C)(C)C)N1C(C(=O)NC2(C(=O)N(C)C)CC2)(COC)C=CC1 c1(C(c2nc(Cl)sc2Cl)C)cccc(OC(F)F)c1.C(C(=O)O)OC Cc1ccnc(C(=O)NCC2CCN(C(COC(C)C)C(=O)OC(C)(C)C)CC2)c1 c1(C(N(C2CCN(C(c3ncn(C(C)C)n3)=O)C2)CC#C)=O)cccnc1 C1(C2CC2)(CNC(CC2(OC)CC2)=O)CCN(C(=O)C(C(C)C)N(C)C)C1 c1(CNC(C2(CNC(C=NOC)=O)CC23CCC3)=O)cnc(O)c(F)c1 c1(NCC(C(C)(C)C)NC(C23CCCN(CCC2)C3)=O)nccc(S(C)(=O)=O)n1 N1(C(CC)=O)CCN(C(C2(C(F)F)CCOCC2)=O)CC1c1nccn1C C(=O)(CC(C(F)F)n1cccn1)N1C2C(NC(C(C)SC)=O)C(C2)C1 N1(C(CC=CC)=O)CCC(C2CCC2)(CNC(=O)CC2CCCCC2O)CC1 C1(CNC(CC2(OC)CC2)=O)CCCC12CCN(C(c1ccc(F)c(Cl)c1)=O)CC2 CCC(C)(C#N)C(=O)N1CCCOC(CNC(c2cnc(C(F)(F)F)s2)=O)C1 c1(CC(=O)NC2CC2NC(=O)CN2CCCC(C(F)(F)F)C2)cc(F)ccc1F c1(CC(=O)NC2CN(C(C(C)(C)OC)=O)CC2O)cc(F)cc([N+](=O)[O-])c1 Cc1cc(C(=O)NC(CC(C)C)c2nc[nH]n2)nc(CO)n1 Cc1ccsc1C=CC(N1CC2CC2(NC(C2CC2c2ccn(C)c2)=O)C1)=O c1(CC)cccc2[nH]c(C(=O)NCCCn3cc(CCN4CCOCC4)nn3)cc12 C1(CN(C(=O)C(N)=O)C)CCN(C(=O)C(C(=O)OC)c2ccccc2)CC1 N1(Cc2cc(C)nn2C)C2CCC1CC1(C2)OCCO1.C12CC(C1)C(=O)N2 c1(NC(c2c(CNC(=O)CC3COCCO3)nccc2)=O)ccnc([N+](=O)[O-])c1 N1(C(=O)OC)CCCC(C(N2CCC(O)(CNC(c3nccnc3C)=O)C2)=O)C1 C12(NC(C(C(C)C)n3ccnc3)=O)CCC(CC1)N(C(C1CCCN1C)=O)C2 c1(C(N2CCC(CNC(C(C)SC)=O)C(F)(F)C2)=O)cc(S(N)(=O)=O)ccc1O C1(CC)CN(C(C2CCC(NC(=O)C3=CCCC3C)C2)=O)CCC1CO c1(OCC)ccc(F)c(C(=O)NC(C)CNC(c2ccn3nccc3n2)=O)c1F c1(OC(c2noc(Cc3ccccc3Cl)n2)C)cc2c(F)c(F)cc(F)c2[nH]1 c1(C(N2CCC2C2CCCCO2)=O)cccc(F)c1.O=C1CC2(CC2)N1 C(=O)(C(C)CC(=O)NC1CC(NC(=O)COC2(C)CCC2)C1)OC C(=O)(C(C)CC(=O)NC(C)CC1CCN(C(c2nccc(Cl)c2F)=O)CC1)OC CC1CCN(c2ncc(O)cn2)C1CNC(C1(C)CC=CC1)=O c1(N(C2CCSC2)C)ccc(S(=O)(=O)N(C2CCCC2)C)c(Cl)c1 C(=O)(C(C)CC(C)C(C)=O)N1C(CC)C(NC(c2cncn2C(C)C)=O)CCC1 CCC(CC)CCC(=O)NC(C1(O)CCCCC1)C(=O)NCc1cccnc1OC N1(Cc2n(C(C)C)nnn2)CC2(C1)SCCC2NC(C1CC12CC2)=O c1(C(=O)NC(CNC(C=NOC)=O)C2CCC2)cc(Cl)cc(N)c1OC c1(C(=O)NCC2CC(OCC)C2)ccc(NC(=O)CNC(=O)C(C)(C)C)s1 c1(OC(C)C(N2CC3(CC3C(=O)Nc3cncc(Br)c3)C2)=O)cc(Cl)ccc1Cl CC1CCC(C(=O)N(CCCC(=O)NC2(C(C)O)CC2)C)CC1 C(CN=c1cc(F)nc[nH]1)NC(C(N1CCN(C)CC1)C)=O C1(C)(CNC(Cc2cn(CC(C)C)nc2)=O)CCCN1C(C1CNC(=O)N1)=O C(=O)(C1CCCc2ncnn21)NCC(CC(C)C)NC(=O)C#CC1CCOCC1 c12ccc(s1)S(=O)(=O)NCC(=O)NCC1CCC1NC(=O)C2.CCC(C)OC C1(C(=O)NCCCCCNC(c2c(OC)scc2)=O)CC12CCCOC2 CCCCC(CC(=O)N(C)CC)NC(=O)CC1CC=CC1.C(=O)C(F)(F)F c1(C(=O)NCC23C(CN(C(c4c(CC)ccs4)=O)C2)C3)ccc(N(C)C)cc1F c1(N2CC(CCCCNC(c3cc(C)ncc3)=O)C2)ncc2c(c1C#N)CCC2 C1(NC(=O)Cc2cc[nH]n2)CCC2(CCN(C(=O)C(O)CC(F)(F)F)C2)C1 c1(NCC(N2C(C)(C(N(CCC)CCOC)=O)CC2)=O)cn(C)nc1C N#CCCCC(=O)NC(CC(=O)N1CC(N2CC(F)C2)C1)C1CC1 CCCN=C(NCCc1cccnc1)NCC(C)CSc1cccc(Cl)c1 C#CCC(C(=O)N1CC2CC1(CNC(=O)C(C)n1ccnn1)C2)SC C1(NC(C2(C#C)CC2)=O)CN(C(C2CN(C3CCOCC3)C2)=O)CC(C)(C)C1 N1(C(CCN(CC#C)C(c2[nH]ccc2C)=O)=O)CCN(C)C2CC12 CC(CC(=O)N1CCC2(CC1)CC2CNC(C1(O)CC1)=O)C(C)(C)C N1(C(C=C(C)Cl)=O)CCN(C(=O)CC(C)C2CCCC2)CC1CO N1(C(COC(C)=O)=O)CCCC(n2cc(CC(N3CCCC3)C)nn2)C1 c1(CC)c(C(=O)NCC(C)NC(=O)Cc2cscc2Br)cccc1F N1(C(COCCC)=O)CC(C)(CCC(=O)NC(C)Cn2cccn2)C1 CCC(CCC(=O)NC1(c2nc[nH]n2)CCC1)NC(c1n[nH]cc1C)=O c1(C(N2C(CNC(CC=C)=O)CCC2)=O)ccccc1OCC(=C)C c1(C(=O)NCC(C)N(C)C(c2ccc(Cl)o2)=O)cc([N+](=O)[O-])c2ccccc2c1 C1(C2CC2)(NC(C(C2CCOC2)NC(C(C)C2(O)CCC2)=O)=O)CCCC1 CN(C)S(=O)(=O)N1CC(C(N2CCC(O)(CNC(c3ccc(=O)oc3)=O)C2)=O)C1 N1(C(C(CC)=CCCC)=O)CC(CNC(C2(n3cccn3)CC2)=O)C(O)C1 c1(C(=O)NC2CC(NC(=O)Cc3cnccn3)C2)ccc(F)c(C(F)(F)F)c1F C(=O)(C1=C(Cl)CCC(C)C1)N(C1CCC(NC(c2ccc(C#C)nc2)=O)CC1)C N1(C(=O)CCOCC(F)F)CCC2CN(C(=O)C(F)C3CCC3)CC2C1 C1(NC(CCOC)=O)CC(=O)N(C2CN(C(c3ccc(CO)s3)=O)C2)C1 N1(CC(C)(C)C(=O)NC2COCC2NC(C2(F)CC2)=O)Cc2ccccc2C1=O CCC(CC)CC(=O)N1CCCCC(CCC(=O)N(C(C)CSC)C)C1 CC1=C(C(=O)NC(C)CNC(=O)CCc2nc3ncccn3n2)C(=O)OC1(C)C Cc1cc(C(=O)NCC(C)CNC(=O)C=C2CCCCC2)cc(C)c1O c1(CC(=O)N(C(C)C(=O)N)CCC)ccc(C)nc1.C(CCS(C)=O)CCOC c1(-c2ccc(CN(CC(C)C)C(c3ccncc3)=O)nc2)ccc2c(c1)NCCO2 O=C1CCC(C(=O)NCCCc2cn(-c3ccc(F)nc3)nn2)c2ccccc21 CCCCCOCC(N1CCC1C(=O)NC1CC1COC)=O C1(NC(CSCC#C)=O)C2CCC(C2)C1C(N1CC(N(C)C)C(O)C1)=O c1(C(=O)NC(CN(C(c2c(C)nc[nH]2)=O)CCO)C)ccc(OCCF)cc1 C(C(=O)NCc1ccc(C(=O)NCC(=O)N(C)O)cn1)(C(C)(C)C)OC S(=O)(=O)(c1cccc2cnccc12)NC(c1c2n(nc1)CC(C)CO2)=O N1(C(C(c2ccc(Cl)cc2)C)=O)CC(NC(=O)Cc2cnc[nH]2)C(O)C1 c1(OC)c(C(N2CC(NC(c3cn(C)cn3)=O)CC2C)=O)nc(O)nc1O N1(C(C2CC(SC)C2)=O)CCC2(CCC2)C(NC(c2ccc(C)nc2C)=O)C1 O=C(C=Cc1ccc(F)c(F)c1)NNc1cnnc(O)c1Cl c1(N(C(C)=O)CCNC(c2csc(CSC)n2)=O)ccc(I)cc1 c1(OC)ccc(C(N2CCCCCC2CNC(c2ccc(C)o2)=O)=O)c(Br)c1 CC(C)(C(=O)NCCC1CCN(C(C2CC2(F)F)=O)C1)n1cc(Cl)cn1 c1(-n2ccc(C(N(CCNC(C=C(CCC)C)=O)CCC)=O)n2)ccccc1Cl c1(-c2c(C(=O)Nc3ccc(C(=O)O)c(C(F)(F)F)c3)c[nH]n2)cccc([N+](=O)[O-])c1 Cc1ccc(C=CC(N2CCN(C(C34COCC(C3)C4)=O)C(C)C2C)=O)cc1Cl N1(C(c2c(C)nc(C)o2)=O)CCN(C(=O)C2=C(Cl)CCCC2)CC2CCCCC12 N(C1CCC(NC(c2csc(COC)n2)=O)c2ccccc21)C(C(=O)NCC)=O c1(OC)cnc(C(=O)NC(C)C(CO)NC(=O)CC(C)(C)C2CC2)c(F)c1 C12(C(N(C3CC(NC(=O)COCC4CCCO4)C3)C)=O)CC1CNC2=O C12(C(N3CCC(N(C(CSCCC)=O)CCC)C3)=O)CCC(CF)(CC1)CC2 CCC(C)C(O)C(=O)NC1CCN(C(c2ccc(O)cc2)=O)C1C(C)(C)C C1(CCC)CN(C(=O)CN2CSCCSC2)CCN1C(c1cn(C(F)F)cn1)=O c1(C(C(=O)NC(CC)C)N(C)Cc2cc(Cl)cc(Cl)c2)cn2cc(Br)ccc2n1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(NC(=O)C(F)(F)c2ccccn2)C(F)C1 c1(C(N(C2CCCN(C(Cc3cnc(C)o3)=O)CC2)C)=O)cc2cccnc2o1 CS(=O)(=O)c1ncccc1NC(=O)NCc1ccn2ccnc2c1 C(=O)(CCCC(=O)NC(C1(CNC(c2cnn(C)c2C2CC2)=O)CC1)C)OC CCC(C)(CO)C(=O)NC1CC(C(=O)NC2CCC3(CC3)C2)CC1O c1(C(=O)NCC(CNC(C(C)N2CCC2)=O)F)cnc2n1CCCC2 N1(C(CNC(CC)=O)=O)CC(C(N2CCC(C)(C3CC3)C2)=O)C(C2CC2)C1 O=C1CCC(=O)N1CCCCCN1CCCC(Cn2ccnn2)C1 N1(C(C2N(C(c3cc(OCC)no3)=O)CC2)=O)CCC(C(=O)OC)CC1 N1(C(c2nc(CCC)sc2)=O)CCOC(CCNC(C2CC2(C)CC)=O)C1 c1(N2CCC(N(CCC)C)C2)cc(C)[nH]c(=NCCN2CCC(OC)C2)n1 CCC(F)(F)CC(=O)NCCC(O)C(=O)N1CCCC(C(F)F)C1 Cn1ccc2ccnc(C(N3CCCC4CN(C(C5(CF)CC5)=O)CC34)=O)c12 C1(NC(CN(CCOC)C)=O)CCC2CCN(C(c3ccc(Cl)c(F)c3O)=O)C12 C1(NC(COc2ccc(OC)c(C)c2)=O)CN(C(=O)C(N)=O)C2(CCOC2)C1 C(C(=O)NCC1(C)CCCN1C(c1ccc[nH]1)=O)(C(C)C)NC(C)=O C1(NC(C2CC(C)N(C)C2)=O)(CO)CCCN(C(c2coc(O)n2)=O)C1 C1(O)(C(=O)Nc2cn(CC)nc2)CCN(Cc2ccnc(C3CC3)c2)C1 c1(OCC(=O)NCCCC(C)NC(C(CCC)N(C)C)=O)cccc(Cl)c1Cl CC(C)CCN=C(NCC12CC1(C)C2)NC1CC(F)(F)C1.OC C(C(C)C(=O)NC(C(c1ccccc1)OC(C)=O)=O)N(C(=O)C(C)(C)O)CCC#N n1(C(C)C)ncc(C(=O)OCCc2ccnc(CO)c2)c1C1CC1 N1(C(Cc2cc(OC)c(F)cc2)=O)CCCC2C1CCN2Cc1nc(Br)cn1C c1(C(N(CC(C)NC(=O)C(C)n2ccnn2)CC)=O)cccc(C)c1Cl O=C(C1c2ccccc2CN1Cc1ccccc1OC(F)F)N(CCO)CCO c1(C(=O)NCC(CC=C)NC(=O)C(C)=C(C)C)ccncc1C=C CC1CN(C(c2coc(C3CC3)n2)=O)CCC1NC(C1CCC(=O)CC1)=O C1(NC(C2CCN(c3cccc(N(C)C)c3)CC2)=O)CSc2nccn2C1 C(=O)(C(CC)CCCCC)N(C1CCS(=O)(=O)C1)C1CN(C(C(CC#C)(C)C)=O)C1 S(=O)(=O)(c1ccc(Br)cc1NCC1NC(=O)CC1(C)C)NC(C1CN(C)C1)=O N(C1CCc2ccc(F)cc21)c1cc(N2CCCCCC2)nc(C(F)(F)F)n1 N1(C(=O)NC2C(C)(C)NCC2)CC(N)CC1(C)C C12(NC(CSCCC#N)=O)CC(NC(c3occc3F)=O)(C1)C2 N1(C(C(c2ccc(OC)cc2)OC)=O)CCc2c(NC(C)=O)n[nH]c2C1 c1(OC)ncccc1C(=O)NC(C)CNC(c1ccoc1I)=O c1(N2C(C(=O)Nc3ccc(C(N)=O)nc3)CCC2)ncnc2c1CCCC2 c1(NC(C(C2C(C)C2C)N(CC(c2cc(C)on2)(C)C)C)=O)ccccc1C N1(C(c2c(C)nsc2)=O)CC2CC1CCC2NC(c1cc(C2(C)CC2)n[nH]1)=O C1(CC)CN(C(=O)C(c2cn(C)nn2)NC(c2ccc(N)cn2)=O)CCCO1 Cc1nc2cncc(C3CCN(C(=O)Cc4csc(C(C)(C)C)n4)CC3)c2[nH]1 C1(NC(C(C(C2CC2)OC)(F)F)=O)CCN(C(C)C)C12CCC2 C12(NC(C(C3CC3)OC)=O)CC1CN(C(=O)CCCc1ccccn1)C2 C(=O)(CCN(OC)C(=O)c1ncoc1CCCC1CCC2(CCC2)O1)OC c1(C(=O)NC(C2CCCCN2C(=O)COC(C)(C)C)C)ccc(N(C)C)nn1 C(C(O)C(=O)NCC1CCOC1=O)NC(C1C(C#N)C1)=O N1(C(C2(COC)CC2)=O)CCC(C(=O)N2CCC(CO)(CO)C2)=C(F)C1 N1(C(CC(C=C)C)=O)CCC(C(N2CCC(F)CC2)=O)(CC)CC1 CCCCCC(CC)C(=O)N1CC2(CC2)CC1C(=O)NCc1nc(C)cs1 C(=O)(CCC(CC)CCC)N1C(CNC(C(C=CCCC)O)=O)COCC1 c1(C(N2CC(CNC(CC3ON=C(CC)C3)=O)(COC)C2)=O)cc(O)nc(O)n1 c1(OCC)nccc(C)c1C(=O)NC(C)CC(C)NC(=O)CSc1ccncc1 n1(CCN(C(C2(CCCC)CCC2)=O)CC)ccc(C(N2CCCC2C(C)CC)=O)c1 C1(C(=O)NCC(C)N(C(c2nccc(C)n2)=O)C)CCc2cncn2C1 C1(NC(COCC=C)=O)CCCCN(C(=O)CC2CC(OCC)C2)C1 C(=O)(C1=NNC(=O)CC1)NCC1C(C)CCCN1C(=O)CC(=O)NC1CC1 C1(C(N2CC(C)(CC(=O)Nc3c(C)nns3)C2)=O)CCc2nc[nH]c2C1 C1(C(N2CCC(n3cc(Cn4c(C)cc(C)n4)nn3)C2)=O)CN2CCCN1CC2 CCCCCCCC(F)C(=O)N1CCCCC1CNC(C1CN(C(C)=O)C1)=O N1(C(C(=O)NC)=O)CCC2(CC1)CN(C(c1cnnc(C)c1)=O)CC(C)O2 C1(NC(c2cc(CC)no2)=O)CC2CN(C(c3c[nH]nc3S(N)(=O)=O)=O)CC2C1 c1(NC(=O)NC(c2ccnc(C)n2)CC)ccc(Br)c([N+](=O)[O-])c1 c1(CNC(c2cc(CCNC(C(CC)CN(C)C)=O)on2)=O)ccc(O)c(F)c1 c1(CN(C)C(C2(F)CCN(C(c3ccc(CO)o3)=O)CC2)=O)ccc(Cl)cc1Cl N1(C(C2C(NC(C3(C(=O)N(C)C)CC3)=O)COC2)=O)CC2(COCC)CCC1C2 CC1(NC(C2CNCC2C2CC2)=O)CCC2(CC1)CC2 C1(N(C)C(c2ccco2)=O)CC2CCC(C1)N2C(=O)Cc1ccc(Cl)cc1F C(C(CC(=O)N1CCC1Cn1cc(CC(CO)CO)nn1)C(F)(F)F)N(C)C N1(C(c2c(CC)cco2)=O)CCCC2C1CCCN2C(c1n[nH]cc1Cl)=O N1(CC)CCC2C(CCN2C(c2cc3cnccc3[nH]2)C(=O)NCCCF)C1=O N1(C(c2n(C(C)(C)C)ncc2)=O)CC(NC(c2ncccc2O)=O)CC(O)C1 N1(C(c2c(C(N)=O)cccc2)=O)CCC2CN(C(C3CNC(=O)C3)=O)CC2C1 c1(NCCc2c(OC)cccc2Cl)cc(Br)ccc1S(=O)(=O)NCC1CCCO1 N1(C(C=CCNC(c2nc(C)c(C)s2)=O)=O)CCC(F)(F)CC1C N1(C(C2OCC(C)C2)=O)CCC2(CN(C(=O)C(C)O)C2)C1 c1(SC)cc(C)c(C(=O)NCCC(O)CNC(=O)C(CN(C)C)N(C)C)o1 C1(NC(C2C(C(=O)OC)C2)=O)CC1C1CCCN(C(C2CSCN2C)=O)C1 C(C(C(=O)N1OC2CCC1CC2)OC)NC(c1ncn(CC)n1)=O Cn1cnc2sc(C(=O)NC3(C)CN(C(C4CCCCNC4=O)=O)C3)cc12 C(C(CC)(CC)NC(C1CN(C(C)=O)C1)=O)NC(C(C)OCCCCCC)=O C(C(N=c1nc(O)c2c(ncn2C)[nH]1)C1CCCCC1)NC(C(C)=CC1CC1)=O N1(C(c2c(N)ccc(Cl)c2)=O)CC2(CCCN(C(C3(CO)CCOCC3)=O)C2)C1 C1(C2CCCC2)(C(=O)NC(CNC(c2cc(C)nc(C)c2)=O)C2CC2)CCC1 c1(CC(C(=O)NCc2n(C)nc(-c3ccccc3)c2)N)csc2ccccc12 C(=O)(C(C1(O)CCC1)NC(C1CCC1)=O)NCCOCCCC c1(C(N(C(CCC(=O)OC(C)(C)C)C(C)(C)C)C)=O)cc2c(cc1O)OCO2 c1(CNC2C(C(=O)NCCc3ccc(O)cc3)C2)ccc(OC(F)(F)F)c(Br)c1 c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NCCC(C)(C)CNC(C1CC(C)C1)=O c1(C(=O)NC2C(CNC(C(c3cccc(C)c3)O)=O)C2)cc2ncccc2cc1Cl C1(NC(c2c(SC)nn(C)c2)=O)CCC2(CC1)CCN(C(=O)Cc1ccco1)C2 N1(C(c2nnc(C)s2)=O)CC2CC(NC(C3CCS(=O)(=O)N3C)=O)C1C2 C1(CC(=O)NCCN(C(C(C)OCCOC)=O)CC2CC2)CC(C)(C)CCO1 CCC(C)C(C(=O)N1CCCC(C(=O)N2CCCN2C(C)=O)C1C)OC N1(C(c2c(C)cc(CC)o2)=O)CCC(O)C(NC(=O)Cc2cccc(C)c2)C1 CC1=C(C(=O)NCC(C)(C)CCNC(=O)CCNC(N)=O)Cn2nnnc2N1C CC1CCC(O)(C(=O)NCC(CO)NC(=O)COc2cc(Cl)cc(Cl)c2)CC1 c1(CSCC)ccc(CN(CC(=O)NCCCCCNc2n[nH]cc2COC)C)cc1 C#Cc1cccc(C(N2CCCC(CC(=O)N(CCC3CC3)C3CC3)C2)=O)c1C.CC CC1(C)CC(NC(c2cc(N)ccn2)=O)CN(C(C23COCC2C3)=O)C1 c1(OC)ccc2c(C(=O)NC3(C)CCN(C(c4ccc(C)cc4)=O)C3)c[nH]c2c1 c1(OC)ccccc1CCCNCC1(O)CSC1 C1(NC(C2(O)CCCCC2)=O)CN(C(=O)COCC2CCCO2)CC12CC2 C1(C(N(C)CC2CC(=C)C2)=O)N(C(c2cscn2)=O)CCCC1(C)C c1(CNC(C2C(CNC(C(CC)OCC)=O)OCC2)=O)cccc(C)c1C CC1N(C(=O)CC(N2CCC(O)(OC3C4CCCCC34)C2)=O)CCOC1(C)C N(C(=NCC(F)F)NC1C(F)(F)C12CC2)Cc1cccc(OCCOC)c1 N1(C(c2c(C)cc(CC)o2)=O)CC2CC(NC(=O)CSc3n[nH]c(C)n3)C(C2)C1 Cc1cc2[nH]c(=O)c(-c3nc(-c4ncnn4C)no3)cn2n1 N1(C(C2CC(C(N)=O)C2)=O)CCN(c2cnc(C(C)O)s2)CC1 c1(C(N(CC(O)COCCCN=[N+]=[N-])C)=O)ccc2nccn2n1 Cc1cc(N2CCN(C)C3(CC3)C2)nc(=NCCCCC(F)(F)F)[nH]1 c1(C(N2CC(NC(c3cnc(C)s3)=O)C(F)C2)=O)cccc(I)c1Cl c1(C(=O)NC(CNC(C(C)OCCC=C)=O)C)cc(F)ccc1OCC#N n1(-c2cn(C(C)(C)C)nc2)nc(-c2ccc(N)cn2)nc1CC1=CCCC1 C1(NC(c2c(C)oc(C(C)(C)C)c2)=O)CN(C(=O)C(C)C(F)F)C2(CCC2)C1 N1(C(Cc2n(C)ccn2)=O)CC2CCN(C(=O)Cc3cn[nH]c3)C(C2)C1 c1(C(F)(F)F)n[nH]c(=NCCCNC(c2cccc3nccn23)=O)o1 CCCCC(C)C(=O)N(CCCNC(=O)CC1CC(C)C1)C c1(SC)ccc(C(=O)NCC2CC(NC(C3CC4(CC4)CO3)=O)C2)cc1 C1(NC(=O)Cn2cnnc2)CC2CCCC(C1)N2C(C1CC2C=CC1C2)=O N1(C(CCC(C)NC(=O)CC23CCC(CC2)C3)=O)CC2CC1CS2=O N1(C(C)=O)CCC(F)(NC(=O)C(n2cc(-c3nn(C)cc3C(N)=O)nn2)C)C1 C1(C(C)C)(CO)CCCN(C(c2ncsc2Br)C(=O)NC2CCCC2)C1 CCC(C)CC(C)C(=O)NCC1(NC(c2ccccc2[N+](=O)[O-])=O)CC(OC)C1 c1(OC)ccccc1C(=O)NC(C)CC(=O)NCCCn1cnnc1 C1(NC(=O)C(O)CCCNC(C23CC(CO)(C2)C3)=O)CCCC2(CCC2)C1 CC(C)(C)C(CO)C(=O)NC1CC(CO)C1 O(NC(=O)C(C)(n1cccn1)C1(CO)CCC1)C(CCC(=O)OC)=O CC1CC(F)CN1C(C1CC(NC(=O)C(C)Cc2cn(Cc3cnns3)nn2)C1)=O CCC(C)C(CNC(C1(COC)CN(C(c2c[nH]nc2Cl)=O)C1)=O)OC n1(CC(=O)OCC)nc(C)c(NC(=O)C(C(C)C)N2CCN(C)CC2)c1C N1(C(C2CC(CC)OCC2)=O)CCCC(C)(CNC(c2ccnc(OC)c2)=O)C1 N1(C(CSc2n(CC)ccn2)=O)CCC2(NC(=O)C(C)CC(C)C)CCCCC12 N1(C(C(COC)(F)F)=O)CCC(NC(c2cc(C(C)C)cnc2O)=O)CC(O)C1 c1(C(=O)NCC(C)NC(c2cnn3cccnc23)=O)cnc2ccnn2c1N C12(C(=O)NC(C(C)C)CNC(c3cnn(C4CC4)c3Cl)=O)CCC(CC1O)C2 C1(N(C(COCC)=O)C)CN(C(c2cnc(C)s2)=O)CC12CC2 C(=O)(C(C)(C)C(=O)NC1CCCCC1C(=O)NCC1CN(C)CCO1)OC C(CCCCC(=O)N(C1CN(C(=O)CC2CC3CC3C2)C1)C)N(C)C C(c1ccccc1F)=CCC(N1CC2C(CNC(c3cc[nH]c3)=O)C2C1)=O C1(CC)C(C(N2CCC(NC(=O)OC)C2)=O)CCCN1C(=O)CC(C)OC N1(C(C=CC2N(C(C(C)OCCC=C)=O)CCC2)=O)CCn2nc(C)cc2C1 C12(CNC(C3CC4CC4C3)=O)CCCC(CN(C(=O)CCN3CCC3)C1)C2 CC(C)C(C(=O)NCC(C)C(F)C(=O)NC1COCC(C)(C)C1)C(C)C CCC(C)(C)NC(=O)CC1CC(CNC(=O)CCOCC(C)C)C1 c1(C(N2CC(C(C)NC(c3nccn3C)=O)OCC2)=O)ccn2c1CSCC2 Cn1cc(C(=O)NCCC2CC(NC(=O)CNC(=O)C3CC3)C2)c2ccccc12 CCC(O)C(F)(F)C(=O)NCCC(C)NC(c1nnsc1N)=O CC(C)CC(O)C(C)C(=O)NC1CC(NC(c2cc3ccc(Cl)cc3[nH]2)=O)C1 C1(CNC(CSSC)=O)CCN(C(=O)C(O)CC2CCCCC2)CCC1(F)F C(=O)(CC1=Cc2ccccc2C1)NC1C(NC(CC(CC)C2CC2)=O)COCC1 N1(C(C(C)C2CCCC2)=O)CC=CC1(C)C(=O)N(C)Cc1nnnn1C N1(C(C2(C)CC(=C)C2)=O)C2CCC1CN(C(=O)CCCCOC(C)=O)CC2 C(=O)(C(F)(CNC(=O)CC1=CCCC1)C(C)C)NC(C(=O)OC(C)C)C c1(C(N2CC(O)CC(NC(c3c(=N)[nH]cnc3)=O)C2)=O)ccc2ccccc2n1 C1(NC(C2C(C=C)OCC2)=O)C2CC3CN(C(c4cnn5c4OCC5)=O)C1C3C2 n1(CCC)cc(C(=O)NCC2CCC(C(=O)N(C)C)O2)nn1 c1(C(N(C2CCCN(C(=O)CC3CCCC3)C2)CC)=O)cnc2c(c1)CCCC2 C(=O)(C1=C(Cl)CCCC1)N1CCN(C(CCCC(C)c2ccccc2)=O)CC1 c1(C(N2CCOCC2CNC(=O)C(F)(F)C(F)F)=O)ccc(Cl)c2ccccc12 C(=O)(C1=CCOC1)NCC(CNC(c1n(C(C)C)ncc1)=O)F c1(CNC(c2cc(SC)nn2C)=O)c(F)ccc(O)c1F CCC(CCCC(=O)NC)OC.N1(CCNC(=O)CC23CCCC2C3)CCC(CO)C1 C(=O)(C(F)C(F)(F)F)NC(C1CCCC1)CNC(c1c(CC(=O)OC)cccc1)=O CC1CN(C(=O)CC23CC(C2)C3)CCC1N(C(=O)Cc1csc(Br)c1)C O=C(C(F)C(F)(F)C(F)(F)F)Nc1nccnc1CO.C123CC(C1)(C2)CNC3=O Cc1cc(C(N2CC(NC(c3cc(-c4ccco4)c[nH]3)=O)C3CC23)=O)c(C)n1C C#Cc1ccc(F)c(C(N2CC(CNC(=O)CC3CC34CC4)OC(C)(C)C2)=O)c1 O=C1COC2(CCCN(C(c3ccc(-c4ccns4)cc3)=O)C2)CN1 Cc1c(CC(=O)NCC2CCN(C(=O)CC(C)N(C)C)CC2)ncn1C C(=O)(C#CC1CCCC1)N1C(C)(CNC(CCN2CC(C)(C)SCC2)=O)CCC1 Cc1nc(C(=O)NCCCN(C(c2cc(C)n(C)c2)=O)C2CC2)nn1-c1nc[nH]n1 c1(C(=O)NC(CCC)C2CCCC2)cn(-c2cnn(CCOC)c2)nn1 C1(NC(CC(Cc2cccc(Br)c2)NC(C)=O)=O)CCCC(F)(F)C1O O=S(=O)(c1ccc(F)cc1)N1CC2CCN(Cc3cncc(F)c3)CC2C1 c1(CC)cc(C(c2nnnn2C2CC(C(=O)OC)C2)NCn2cc(C)cn2)n[nH]1 N1(C(Cc2cc(C)on2)=O)CCC(C)C(NC(c2nccn3ccnc23)=O)C1C C12(CC(=O)NC(CC3CN(C(Cc4c(C)nn(C)c4)=O)C3)C)CCC(CC1)CC2 C1(C(N(CC)CC2CC2)=O)CC12CCN(C(c1cc(F)c[nH]1)=O)C2 c1(C(CNC(C(CC2CC2)OC)=O)NC(c2sccc2Cl)=O)cccc(C)c1 c1(CCNC(c2nnnn2C(C)(C)C)C2(CC)CCC2)ccc(SC)cc1 c1(C(=O)NC23CC(C(=O)NCC(=O)OCC)(C2)C3)c(C)ccnc1C c1(NC(C(=O)NC(COC)Cc2cccc(Br)c2)=O)cccc(P(C)(C)=O)n1 CCC(C)(F)C(=O)NCCCCCNC(=O)C(C)Cc1ccc(Br)cc1 Cc1cc(CN2CCOC(CNC(c3cc(Cl)ccc3C)=O)C2)cc(Cl)n1 Cc1cc(C)c2cc(C(=O)N(C3CN(C(C4CC4C4CCCC4)=O)C3)C)sc2n1 C#CCC(CC(F)F)NC(=O)C(C)(C)CNC(=O)C(C)C=C C1(CNC(C=C)=O)CC(F)(CNC(C2CCCN2C2CCCC2)=O)C1 c1(NC(N(C2CCCC2)CCC=C)=O)cnn(-c2ccccc2)n1 c1(C(=O)NC23CC(C(=O)NC4CC(O)C4)(C2)C3)cc2ccccc2cn1 C(=O)(C(C)(C)C(F)(F)F)N1CCC2(C(NC(C=Cc3n(C)ncc3)=O)C2)C1 C1(C(=O)NCC2OCCC(NC(CCC(=O)NCC)=O)C2)CCC2CC1C2(C)C c1(OCC=C)ccc(C(N2CCC3CC23)C(=O)NCCCNC(C)CC)cc1 C(=O)(C1CCCn2nccc21)N1C(COC)CN(C(=O)COC2CCCC2)CC1 C=CC1COCCN1C(C1CCN(C(=O)C(C2CCC2)OCC)C1)=O C(=O)(CCCCC(C)C)N(CCOC(c1n(C)nc(C)c1Br)=O)CC1CC1 c1(C(=O)NC2CC(C)N(C(=O)Cc3ccccc3)C2)cnc2[nH]c(O)nc2c1 N1(Cc2ccccc2)CC=C(C(=O)NCC2CCCCCCN2)CC1 C1(C(=O)NC2CCN(C(C3CC(CC4CC4)C3)=O)CC2)CC12CCOCC2 Cc1c(C(=O)N(C2CN(C(=O)Cn3c(C)csc3=O)CC2F)C)cncc1Cl C(CC(C(=O)NCC1COCC1O)NC(=O)CCCN(C)C)SC C1(CC=C)(NC(c2n[nH]cc2OC)=O)CCN(C(=O)C(c2ccncc2)C)CC1 C1(COC)(CNC(=O)C(C(C)C)SC)CCCN1C(c1cnn(CCF)c1)=O Cc1c(C(=O)NCCC2COCCN2C(=O)C=Cc2cnc[nH]2)cnn1C1CC1 c1(C(=O)NCCN(C(=O)C=C2CCCCC2)C(C)C)nocc1Br N1(C(c2c(C)scc2)=O)CC(NC(c2cnc3n2CCC3)=O)C(C)(C)C1 C1(C)(CC)CN(C(=O)CN(C2CCC2)C(c2coc(C)c2)=O)CCO1 CN1CCC(n2cc(C(=O)NCC3(O)CN(C(=O)CSCC(N)=O)C3)cn2)CC1 c12ncn-1n2.c1(C(=O)NCCN(C(=O)C(=O)NC)CCOC)ccc(COC)o1 CCC1=NOC(C(=O)NC2CC(CCNC(c3oc(C(F)(F)F)nc3C)=O)C2)C1 C1(NC(C=CCCC)=O)CCCN(C(=O)CCc2cc(Cl)no2)C1C Cc1cc(N)c(C)nc1C(=O)N(C)CCN(C(=O)C(F)n1cccn1)C CC(C)(C)C(C)(O)CNC(=O)CNC(=O)CC1CC(=O)NC1=O c1(C2(C(=O)NCC3CN(C(CSCC#C)=O)CC3C)CC2)ccc(F)c(Cl)c1 C1(C(=O)NCCC#N)CCCC1CNC(=O)CNC(c1c[nH]nc1Cl)=O C1(NC(C(C)(C)SC)=O)CS(=O)(=O)CC1NC(c1cccc(C(C)C)c1F)=O C1(C#N)(C(=O)NC2CN(C(CCc3ccc(OC)cc3)=O)C2)CCCOC1 C1(NC(=O)CC2CC2)C2CCN(C(c3cnn(C4CCCC4)c3)=O)CCC12 CCCC(C)(O)CC(=O)N1CCN(C(C2CCNC2=O)=O)C(c2ncc[nH]2)C1 C1(CCNC(=O)CN2CCCCC2)CCCCN1C(=O)CNC1CCCC1 C1(NCCNC(c2n(CCOC)nnn2)C2COC2)CCNC(=O)CC1 c12cc(nn1C)C(=O)NCC2.N1(C(C2CCC(OC)C2)=O)CCCC(C)C1 CSC1=C(C(=O)NC2CCCCC2NC(C2(OC)C=CC=C2O)=O)CCCC1 N1(CC(C(=O)NC(C)C)NC(C2(COC)CC2)=O)Cc2ccc(C)cc2C1 c1(CN(C(C2(C(F)(F)F)CC2)=O)CC)ccccc1OC(F)F CC1(C)C(NC(C2CCOCCN2C(C2CC=CC2)=O)=O)C(C)(C)C1O C1(CNC(CC2(COC)CCCC2)=O)(NC(c2cnc(C)[nH]2)=O)CCCCCC1 c1(NC(C(CC=CC)NC(c2ccc(F)c(F)c2)=O)=O)cccc2c1CCC2 c1(C(=O)NCC(C)CC2CC2)cc(CNC(C2(C)CSC2)=O)no1 C1(NC(CCCCOCCC=C)=O)CCCCCN(C(C2CCS2(=O)=O)=O)C1 C(=O)(C(C)CC#N)NCC(C(=O)NCc1scc(C)n1)O C(=O)(C1CCCc2nc[nH]c21)N1CCCC(NC(c2cccc(N)c2F)=O)CC1 Cc1nn[nH]c1C(=O)NCC1(C(=O)NC(C)C(=O)NO)CCCO1 c1(C(N2C(C)C(NC(=O)CCNC(=O)CO)CCC2)=O)cccc2nc(S)oc12 c1(C(N2CC(C(C(=O)NCCC(=O)NC)O)C2)=O)ncc(C#N)cc1C c1(CC(N2CCC3CN(C(C=C(CCC)C)=O)CC32)=O)oc2ccccc2c1C c1(NC(C(c2ccc(Cl)s2)C)=O)ccc(C(N)=O)nc1 c1(C(=O)NCCCN(C(c2n[nH]c(C)c2O)=O)CC)[nH]c(C)c(S(N)(=O)=O)c1C N1(C(c2scc(OC)c2)=O)CCOCC1CN(C(=O)C(C1CCCCC1)O)C C1(NC(C(N)CO)=O)CCN(CCCc2nccs2)CC1 c1(C(N2CC=CC(NC(CC(C)n3ccnc3)=O)C2)=O)cc2c[nH]cnc-2n1 CC1(C)Cc2ccc(C(N3CCCCC(NC(C4CCO4)=O)C3)=O)c(O)c2O1 Cc1nn(CC(N2CCN(C(c3cncnc3)=O)CC2CCO)=O)c(=O)n1C C1(C)(CSCCOC)CCCC1C.c12ncc(s1)c(=O)n2C1CCCCC1 N1(C(c2c(C(=O)OCC)c[nH]n2)=O)CCC(c2c[nH]cn2)CC1 C=Cn1ncc(C(=O)NC2(CC(N3CCC4C(C(N)=O)C4C3)=O)CC2)c1N C(C(=O)N(C)CCN(C)C(c1cscc1C1CC1)=O)(C(C)C)OCC(C)C c1(C(=O)NCC=CCNC(CC(C=C)C)=O)cnc2sc(C)cn12 c1(CCC)ccc(C(=O)N(C(CNC(=O)Cn2ncnn2)C2CC2)C)cc1 c1(C(N(CCCNC(=O)COC(F)(F)F)CC)=O)cc(CSC2CC2)cs1 Cc1cc(CN2CC3(CC3C(=O)NCCc3nccs3)C2)c(O)c(Br)c1 c1(NCCCCC(C)NC(C=C(C)Cl)=O)cc2c(cn1)C(=O)CCC2 c1(NC(=O)C(N2CCOC(C3CCOCC3)C2)=O)cccc(-c2ccccn2)c1 C1(CCNC(c2c(C)noc2)=O)CC(F)(F)CN1C(=O)CCC1CCC1 C=CC(O)(C(=O)N1CCCN(C(C2CCN(C(C)=O)C2)=O)CC1)C(F)(F)F CC1CN(C(c2ccc(Br)s2)=O)CCN(C(=O)C(F)CC2CCOC2)C1 CC(C)(C)C(C(=O)N1CCC(CCNC(C2(C(C)(F)F)CC2)=O)CC1)C1CCC1 C1(C#N)(C(=O)NCC(CC)NC(C2(Cc3ccccc3)CCC2)=O)CCCO1 CC1(C)CN(C(=O)CN2CCS(=O)CC2)C(CNC(C2(C#N)CC2)=O)CO1 CC1=C(C(=O)NCC(CC2CCCC2)C(=O)N2CC(O)C2)CC1 c1(Cn2cc(C3CCN(C(c4cc(C)[nH]n4)=O)C3)nn2)ccccc1Br c1(C(N(CC(C)NC(C2CCN(C(=O)C3CC3)CC2)=O)C)=O)cc(F)ccc1Cl C(C1c2ccccc2CCN1C(=O)C=CCO)NC(C(C)C1CCC1)=O C1(NC(c2ccc(CC)o2)=O)CC(C)CN(C(C23CC4CC2C3C4O)=O)C1 c1(C(=O)NC(C(C)NC(c2cc(CC)n(CCO)n2)=O)C)ccn2nccc2n1 N1(C(CSCC)=O)C2CCC1CC(C(=O)NC(C)C)C2.C12CC1C(=O)O2 Cc1ccc(C(N2CCC(C(=O)NCC(c3cccs3)C)C2)=O)n1C C1(NC(C2CCOC2)=O)CCCCCN(C(=O)CN2CCOCC2=O)C1 C(c1ccccc1)=C(CNC(CC(C)C(=O)NOCC(C)(C)O)=O)C c1(NC(C2(CNC(=O)CCCc3ccccc3)CC2)C)ccc([N+](=O)[O-])cc1 N1(C(C2CCC(F)C2)=O)CCN(C(c2ccc3c(c2)OCO3)=O)C2(CCC2)C1 Cc1ccnc(N2CC=CC(NC(C3CCCC3O)=O)C2)n1 N1(C(CC=CC(C)(C)C)=O)CCC(C)(C)C1C(=O)Nc1cc(F)ccc1O c1(C(=O)NCCCC(C)(C)NC(c2cccc(N)n2)=O)cnn2ccsc12 C=C(C)CC(C(=O)NCCC(C)O)NC(c1nc(Cl)cs1)=O c1(OC)c(Cl)nc[nH]c1=NCC1CCCC(NC(c2cc3c[nH]nc3s2)=O)C1 Cc1cn2cc(C(=O)NC3(C)CN(C(c4nn(C)cc4C)=O)C3)sc2n1 C1(C(=O)NC2CCN(C(CCc3[nH]c(=N)sc3)=O)C2)CC2CC1CC2O N=c1nc2ccc(C(N3CCOCC(NC(c4sccc4Cl)=O)C3)=O)cn2[nH]1 Cc1cc(C(=O)C(=O)NC2CN(C(C3CCSC3)=O)C2)ccc1F CN1CC(O)CC1(C)C(=O)NCC(C)(C)NC(=O)Cc1cncnc1 Cc1ccc(-c2noc(C34CC(C(=O)OC(C)(C)C)(CO3)C4)n2)c2[nH]ncc12 c1(C(=O)NC(C)(C)CCNC(=O)CC2CC(F)C2)ccc2c(c1)NC(=O)CC2 C(=O)(C1=C(Cl)CCOC1)N1CC(N(C)C(c2ccncc2N=[N+]=[N-])=O)C1 c1(CC)cc2c(NCC3CCC(NC(C4C(C)OC(C)C4C)=O)C3)ncnc2s1 Cc1nc(CC(C)C)oc1C(=O)NCC1(C)CCN(C(=O)CC(C)NC(N)=O)C1 Cc1cc(C(=O)NCC2CCC2NC(=O)CC2NC(=O)NC2=O)oc1Br Cc1nc(CC(=O)NCCC2CCCN2C(c2cc(Cl)no2)=O)sc1C N1(C(CSCC(C)C)=O)CC2(C1)CN(C(c1cncc(Cl)c1)=O)C2 C1(N(C)C(C2(O)COC2)=O)CCCN(C(=O)C(F)(F)c2cnn(C)c2)CC1 C1(C(=O)NC23CC(NC(C(OC)OC)=O)(C2)C3)CC(=O)N(C2CC2)C1 N1(CCCN(C(CC2C(CC)C2)=O)CC(C)C)CCC(O)CC1 N1(C(c2cnc(N(C)C)o2)=O)CC2(C1)CN(C(c1cc(Br)ncc1F)=O)CCO2 C=CC1CCCCN1C(=O)C(C)CCCOC c1(NC(CSCC#C)=O)c(P(C)(C)=O)ccnc1O CCC(C)CC(=O)C(=O)N1CC2CCN(C(=O)Cn3cc(COC)nn3)C2C1 C=CCC(CC(F)F)C(=O)NC(CNC(c1sccc1C(C)C)=O)C(C)C(C)C c1(C(N2CC(C(C)NC(C3CC(C)(O)C3)=O)C2)=O)c[nH]c2cccnc12 CN1CCN(C(=O)C(=O)Nc2ncc[nH]2)C(CNC(=O)CCc2nncn2C)C1 C1(OC(c2c(CCC)[nH]cc2)=O)CCC(S(C)=O)C1 c1(C(C(=O)NCC(C2CC2)SC)NC(=O)CC2OCCC2C)c(C)cccc1Br CCC(C)(C)CCCC(=O)NCCCCC(C)NC(=O)C(c1ccnn1C)C c1(NC(c2ncsc2C(N2CCN(C)CC2CO)=O)=O)nccc2[nH]ccc12 C(=O)(C1=CCCNSC1)NC(CCN(C(COc1ccc(C)c(C)c1)=O)C)C Cc1cccc(C(C)NC(=O)C=CC2CCCN2C(c2ccoc2Cl)=O)n1 c1(SCC)cnc(O)c(C(=O)NCC(CC)NC(=O)CC2CCOC2=O)c1 C(=O)(CC(C)C(C)C)N1CC(CNC(C(C)Sc2nnnn2C2CC2)=O)OCC1 c1(-c2c(CC)noc2)nc(-c2cccc(OC(C)C)c2)nn1C1CCC1 C1(NC(Cc2cnc(C)[nH]2)=O)CN(C(=O)Cc2cccc(C)c2F)CCC1C C1(CC(=O)NCC2C(OCC)C2)CCN(C(C2COC(=O)C2)=O)CC1 C(=O)(CC(O)C(C)C)N1CC(NC(C(c2ccccc2)N(C)CC)=O)C(CC)C1 c1(CNC2(C=C)CCC2)cccc(OCC(=O)O)c1 N1(C(C2C(C)(C)C2CNC(=O)C(N)=O)=O)CCOC(C)(C(N)=O)C1 c1(C(N2CCC(NC(CCCOCCC)=O)C2C)=O)cccc2ccnn12 C12CCC(CC1)C(c1nnnn1C)N2.C1(OC)CC(CC(=O)OC)C1 CC(=O)CCCC(=O)N1CCC(NC(=O)CCc2ccc(F)nc2)C1C c1(C(CNC(CC)C(=O)OC)=O)c(F)cc(Cl)cc1Br c1(OC)ccccc1C(CF)NC(N1CCCC1C(F)(F)F)=O c1(CCCC(=O)NCC2C(CNC(C(CC)F)=O)C2)ccc(Cl)c(Cl)c1 C=CCC(F)(F)C(=O)N1CCN(CC2CN(C(c3cncc(OC)n3)=O)C2)CC1 CCC(F)C(=O)NCC1CCN1Cc1ccccc1.c12ncnn1CC(=O)OC2 CC1(F)CCN(C(C2CCC(CNC(c3cc(C4CC4)no3)=O)O2)=O)C1 C=CC(C)C(=O)N(CCCC(=O)N(CC(C)(C)O)C)C c1(C(=O)NCC2C(NC(=O)Cn3ccc(C4CC4)n3)C2)cc2c(s1)CCCCCC2 c1(C(=O)NC(CNC(CCSC)=O)CC(F)(F)F)c(C(F)F)nc2ccccn12 Cc1nccc(C(=O)NCC(C)NC(=O)CC(C)N2CCCC2=O)c1C c1(CC(=O)NC(C(=O)NC2CC(C=C)C2)C2(C)CC2)cnccc1OC C=CC1(C(=O)NCC(C)(C)CC(C)C)CCN(C(C2CC3(CCC3)CO2)=O)CC1 C1(NC(CNC(CNC(CC)=O)=O)=O)CCCCN1C(c1ccnc(C)c1)=O C1(CC(=O)NCCOCCCN(C(=O)CCc2cnc(O)[nH]2)C)CCC(C#N)C1 N(S(=O)(=O)N(C)CCN1CCCC1CO)CCOC c1(C(N2CC(NC(C(C)OCCCC)=O)C(C)CC2)=O)c[nH]c2cc(C)ccc12 CN1CC2C(C(N3CC4CC3C4C(=O)NC(C)(C)C(F)(F)F)=O)C2C1 c1(C(C(=O)NC(C)CCNC(C2CCC(N(C)C)C2)=O)C)c(F)cccc1F N1(C(C(CNC(C2(OCC)CCOC2)=O)(C)CC)=O)CCOC(C)(C)C1C C12(CNC(CC3(COC)CC3)=O)CCCCC1CN(C(c1cncnc1)=O)C2 C1(NC(C(C)OC)=O)CN(C(=O)CC2(n3cnnn3)CCOCC2)CC(C)(C)C1 c1(C(=O)NCCC(C)N(C(C2N(C(CC)=O)CSC2)=O)C)ccc(S(C)(=O)=O)o1 N1(C(C(=O)N(C)C)=O)CC(C2CCCCN(C(c3c([N+](=O)[O-])cnn3C)=O)C2)C1 c1(OC)nn(C)cc1C(N1CCC(CO)(CNC(C2CC2C(F)F)=O)C1)=O c1(NC(CC2C(CNC(c3c(OC)cncc3)=O)C2)=O)ccc(O)cc1F N1(C(c2cnn(C)c2Cl)=O)CC(NC(=O)CN(C2CCSC2)C)CC1(C)C CCC(CC(F)(F)F)C(=O)NCC1(F)CC(CNC(=O)C(O)C2CCC2)C1 c1(CNC(C2CC2NC(c2cccc(Cl)c2)CO)=O)cc(Cl)ccc1O C1(CNC(CCC(=C)C)=O)CCC(C)(C)CN1C(=O)C(=Cc1cccnc1)F CCC(CN(C)C)CC(=O)NCCCC(C)(C)C(=O)NCCCC(C)(C)CC N1(C(CCNC(COC)=O)=O)CCC(NC(c2coc(C(F)F)c2)=O)C(C)(C)C1 C(=O)(C1=NOC2(CCC2)C1)NCC1(C)N(C(C(CC)O)=O)CC(F)(F)C1 C=CC(CC)CC(=O)NCC1CCCN(C(C2CCCCNC2=O)=O)C1 C=CCCCC(C(=O)N(C)CCOC1CC1)NC(C1CCC(=O)C1)=O C1(NC(C(C2CCC2)NC(c2c(C)cccc2)=O)=O)CC2C(C1)C2(F)F Cc1cnc(C=CC(=O)NCC(C)(C2CC2)NC(c2ncoc2C(C)(C)C)=O)[nH]1 c1(C(=O)NC2CC23CC(NC(C2CC4C=CC2C4)=O)C3)cc[nH]c2nccc1-2 NC1C2C=CC(O2)C1C(N1CC(CCc2cn(CCF)nn2)C1)=O CC1(C)C(C)(C)C1(F)C(=O)NCC1CCCCC1NC(c1coc(CO)c1)=O c1(OC(c2cc(OC(C)C(=O)Nc3cnccn3)no2)=O)ccc2c(c1)CCC2 N1(C(Cn2ccc(C)n2)=O)CCCC2C1CCN2C(c1csc2c1CCCC2)=O C1(CC(=O)NC(c2ccccc2)C#C)CCC(NC(c2ccsc2C)=O)CC1 c1(C(C)CC(=O)NC2(C(=O)O)CCOC2)ccc(F)c(Br)c1 Cc1c(-c2cnn(C3CC3)c2)cnc2c1N(C(c1ncccc1F)=O)CCO2 c1(CC(=O)NCCCCN(C(C(C2CCC2)OCC)=O)C)c[nH]nc1C C1(C(N2CC(NC(c3cc(CC)no3)=O)C(OC)C2)=O)CC(C(C)(C)C)=NO1 N(C)(C1CN(C(=O)CO)CCc2ccccc21)C(c1c(C)cncc1)=O C1(NC(CC2N(CC)CCOC2)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)C(C)C1 CC1C(NC(=O)CC2CCCCC2C)C(C)CCN1C(c1cc(F)cnc1O)=O C1(NC(C=CCC)=O)CCN(C(=O)CC(C)C2CCC2)CC1C Cc1cc(C)c(CCNC(c2ccc(Cl)cc2F)c2nnnn2C2CC2)c(C)c1 N1(C(c2cc(CC)oc2C)=O)CCC(C)(C)C(C(=O)N(c2cccc(Cl)c2)C)C1 C1(NC(C2(COC)CC=CC2)=O)CC12CCN(C(=O)C(C1CCC1)OC)CC2 C(=O)(C1=Cc2ccccc2OC1)NC(CNC(C1C(C)(C(F)(F)F)C1)=O)CO c1(C(=O)NCCN(C(c2cccc(O)n2)=O)CC2CC2)cc2n(c1)CCC2 C(CC)(CCCC(=O)NC1CCNC1=O)NC(C(C=C)(F)F)=O c1(C(=O)NCCC(C)CCNC(=O)CCS(C)=O)ccnc2[nH]c(O)nc12 C(=O)(C(Cn1cccn1)NC(=O)C(F)CC)N1CC(N(CC(C)C)C)C1 C=C(C)C(C)(C)C(=O)N(C1(C(=O)NCc2ccc(C#N)s2)CC1)C Cc1cc(CN2CC(C(=O)Nc3cn4ccsc4n3)CC(F)C2)c(O)c(Br)c1 N12CC(C3(CC3)C1=O)C2.N1(CC(N2CC(CC(C#C)C)C2)=O)CCN(C)CC1 N1(C(c2cncc(C)c2)=O)CCC(CNC(=O)Cn2cccc2)C(C)C1 C(C)(CCCCN)NC1CC(CO)C1.C=CC(C(=O)N)OC c1(C(N2CCC(C)(C(=O)NCc3cccc(Cl)c3O)C2)=O)nccc2[nH]ccc12 N1(C(CSCC)=O)CCC2(CCCN2C(c2cc(O)ccc2Cl)=O)C1 Cc1ccncc1CNC(=O)CC1CN(C(C2CC2(C)C)=O)CC1C C1(C(=O)OC)C(F)(F)C12CC(C(=O)N(CCCNC(C1(CO)CC1(F)F)=O)C)C2 C(=O)(CC1=CCCCC1)NC1C(CC(=O)NC2CC(O)C(O)C2)CCCC1 C=CC1(CC(=O)NC(C)CCSC)CN(C(=O)CC2COCCOC2)C1 c1(C(N(CCCNC(Cn2ccc(C)n2)=O)C)=O)ncc(Br)cc1F C1(CNC(=O)NCc2nc(CC)[nH]n2)CCC(=O)NC1C C(CC(C)(C)C(=O)NCCCN(C(=O)CNC(=O)NC1CCCC1)C)NC(C)=O c1(C(N2C3(CN(C(=O)CCn4cccnc4=O)C3)CC2)=O)noc2c1COCC2 Cc1nncc(C(=O)NC2CC3(C2)CC3NC(c2ccncc2N(C)C)=O)c1C CCCC(CC(=O)NCCN1CCCC2CC12)NC(C1CC2CCCC2C1)=O CC(O)C1CCCc2ccccc2C1NC(=O)C(N1Cc2ccccc2C1=O)C C1(N(C(C2(F)CN(C)C2)=O)CC)C(CO)CCC12CCC2.C12(C(=O)N)CC3CC1C2C3 C(=O)C(C)C(O)CC(C)C.CON(CCO)C(=O)CON c1(C(N2C(CNC(CC=C)=O)CCCCC2)=O)c[nH]c2ccc([N+](=O)[O-])cc12 N1(C(CC)CO)CCN(C(c2csc(C(C)N)n2)=O)CC1 c1(C(N(C2CN(C(=O)C=CC=C(Cl)Cl)C2)C)=O)ccc(F)c(N)c1 c1(C(N(C)CC2CCN(C(C3(C#N)CCOC3)=O)CC2)=O)c[nH]c2cccnc12 CCC(CCCC(=O)NCC#CC(F)(F)F)NC(C1C2CCCC(=O)C12)=O N1(C(CC2N(C)C(=O)CC2)=O)CCCC(C)(CNC(C2(C3CC3)CCC2)=O)C1 N1(C(C(CCC)=CCC)=O)CC(C)C(C)(C(=O)NCCCN2CCCC2C)C1 c1(C(=O)NCC(C)(CO)NC(CS(CC)=O)=O)cnc2ccc(C)cn12 n1(CC(=O)NC2COCC2CNC(C2(n3cncn3)CC2)=O)ncc(Br)n1 CC1(C)CC(CC(=O)NC(C2CCCO2)CO)N(C(=O)C=Cc2cscn2)C1 C(=O)(N=c1cc(C(=O)N(C)C)n(C)[nH]1)NC(C)C(F)(F)F C(=O)(CCCCC(=O)NC1(C(=O)NCCC2=CCCCC2)CCOCC1)OC c1(CNC(C(C)NS(=O)(=O)C(F)(F)F)=O)ccc(Cl)c(Cl)c1F C1(CC)(CCN(C(CNC(=O)Oc2ccccn2)C)C)CCOCC1 C(=O)(C(C(C)C)C(C)C)N(CCC(C(C)(C)C)NC(C(C(C)C)OC)=O)C C=CCCCC(C(=O)N1CC(CC)(CO)C1)NC(=O)C=CCO c1(NC(C2CCN(Cc3cn(C4CCC=CCC4)nn3)C2)=O)ncc(Cl)cc1F C(=O)(CCS(N)(=O)=O)N(C1CCCCCC1)CC(=O)NCC1(O)CN(C)C1 c1(C(N(CCNc2cc3nc(C)ccc3o2)CC)=O)c(Cl)oc2ccccc12 Cc1cnc2n1CCC(C(=O)NCCCn1cc(-c3ccccn3)nn1)C2 Cc1cc(C(=O)NC2CCC(N(C)C(C3(CO)CC3(F)F)=O)CC2)ncn1 C(CCF)(C(=O)NCc1ccns1)NC(C=CC(=O)OCC)=O C1(NC(C2C(OC(C)=O)C2)=O)CC=C(C(=O)N2CCN(C)CC2CO)C1 O(NC(=O)C(CNC(=O)COc1cccnc1)CC1CC1)CC(=C)C c1(OCCOCC=CC(=O)NC(C)CNC(=O)Cc2cnc[nH]2)ccccc1 C1(NC(C2N(C(CCC=CC)=O)C(C3CC3)CC2)=O)CC2(CCCCO2)C1 Cc1cc2c(C(=O)NC(CO)CC(F)F)nccn2n1 C1(C(=O)NCc2ccc(Cl)s2)CC(F)CN(Cc2ccc(C(F)(F)F)c(F)c2)C1 N1(C(Cc2c(C)noc2Cl)=O)CC2(CCCN(C(c3cc4c(nn3)CCC4)=O)C2)C1 N1(C(C2CC3CCC3C2)=O)C2CCC1CC(NC(C1CC(n3cnnc3)C1)=O)C2 c1(C(=O)NC(C(C)NC(c2ccc[nH]2)=O)C)c(F)ccc2occc12 N1(C(=O)NC(CC)C(F)F)CCc2ncnc(N(C)C)c2C1 C1(C(N2CC(CN(C)C(C3C4CCOCC34)=O)OCC2)=O)C2(CCC2)C12CCC2 C(C1CCCn2ccnc21)NC(c1ccc(F)nc1)CCl N1(C(C(C)O)=O)CC(CO)C2(CCN(C(=O)Cc3nccn3C)CC2)C1 C1(C(=O)NC2C(n3cc(CCCS(C)=O)nn3)CCC2)CCC(=O)CC1(C)C C1(C(CO)NC(=O)C=CC2CCCO2)CC2(CCC2)C1 CN1CC(C(=O)NC2CC(CNC(=O)C(N)=O)C2)C(C(F)(F)F)C1 N1(C(CC(C)OC)=O)CC2CCN(C(=O)C(C)CN(C)C)CC12 C(CNC(C1CCC(=O)C1)=O)(C(=O)N(C)CC1CC(O)C1)OC CC1=C(C(=O)N2CC(CNC(=O)Cc3conc3C)CC2C)CCS1(=O)=O C12(C(=O)NCCN(C3CCCC3)C(c3n(C)ncc3Br)=O)CCC(CC1)CO2 C(=O)(CCOCCOCCN(CCCN)C)N(CCC1CC1)CC C(N=c1[nH]cnc(SCCCCS(C)(=O)=O)c1C)c1c(C)ccs1 C1(CCNC(C2(COC)CC2)=O)CN(C(c2cccc[n+]2[O-])=O)CCCO1 N1(C(C23N(C(C(CC=C)NC(C)=O)=O)CC(C)(C2)C3)=O)CCCN(C)CC1CC C1(C)(C(=O)NCCCN(C(C(C)CC(N)=O)=O)C2CC2)COc2ccccc2O1 N1(C(=O)CC2CCC=CCC2)CC2CCN(Cc3ncccn3)CC2C1 C1(CCC)CN(C(=O)CC(C)C)CC1C(=O)NC(C)(C)CC Cn1c(=O)ccn(CC(=O)NCCCC2CC3CCC2C3)c1=O n1(CC)nnc(C(=O)NCC(C)(C2CC2)NC(=O)Cc2cc(C3CC3)on2)c1C O=C(CCC(=O)NC1CC1NC(c1cc2occc2[nH]1)=O)NCc1ccccc1 C(=O)(C(C)CSC)N1CC(C(C(=O)NCCC2CCOC2)OC)C1 C(=O)(CC(=O)NCCC1CCCN1C(=O)CC1(O)CCOC1)NCC#C S(=O)(=O)(c1c(Cl)cccc1Cl)N(c1nc(SC)c(F)cn1)C1CCNCC1 c1(C(C)C)ccc(C(N2CC3C(CNC(C4C5CC6C(C5)C46)=O)C3C2)=O)cn1 c1(NC(C23C(CN(C(=O)Cc4ccc(F)cn4)C2)C3)=O)c(Cl)cnnc1Cl N1(C(C=Cc2n(CC)ncc2)=O)CCC(O)C(NC(C2(O)CCSCC2)=O)C1 C1(CNC(C(C=C)OC)=O)CCC2(CN(C(=O)CCCC3OCCO3)C2)O1 C1(NC(CCc2nc(C)sc2)=O)CCC(CC(=O)Nc2ccccn2)CC1 N1(C(C(CC(C)c2ccccc2)C)=O)CCN(C(=O)Cc2cc[nH]c2)CC(O)C1 Cc1cocc1C(N1CC(F)(CNC(=O)C(C)N2CCC2)C1)=O c1(COC)cc(C(=O)NC2CC2NC(c2ccc(C(=O)OC)s2)=O)no1 C(=O)(C(=O)C(C)C)NC1CCNCC1N(c1nnc(OC)o1)C(C)=O c1(COC)cc(C(=O)NCC2(CNC(=O)CC3CC4C=CC3C4)CC2)c(Cl)cn1 c1(C(=O)NCC(CNC(CNC(CCC)=O)=O)F)nnn(C)c1CC C=CCCC(C)(C)CNC(=O)CN(C(=O)CCCCC1CC1)C1CCC1 S(=O)(=O)(c1cccs1)NC1C(C(N2CC(C(N(C)C)=O)OCC2)=O)C1 c1(C(=O)NC2C(C)CN(C(=O)C(=O)C3CCCC3)CC2)cc2n(n1)CCCO2 Cc1cc(OCCCC(=O)NC2CC(NC(c3ccnc(S)c3)=O)C2)ccc1Cl CC(Cc1ccccn1)C(=O)NCC(C)(CO)NC(=O)C=Cc1ncc[nH]1 c1(C(CC)C(=O)N(C(C)CNC(=O)Cn2cccn2)C)ccc(Cl)cc1 c1(C(=O)NCC2C(C(=O)NC(c3ccccc3)C#C)C2)cnccn1 Cc1c[nH]c2ncc(C(=O)NC3COCC3NC(c3ccn(C)c3)=O)cc12 C1(CCNC(C(CC)=CCCC)=O)CCN(C(=O)CNC(=O)C2CC2)C(C)C1 N1(Cc2nc(C(=O)O)sc2)CCC2(CN(C(c3cccc(C4CC4)c3)=O)C2)C1 N1(C(COC)=O)CCN(C(C2CC2c2ccc(F)cc2)=O)C(CS(C)(=O)=O)C1 c1(C(=O)Nc2ncccc2Br)[nH]nc2c(-c3cncs3)cccc12 C1(NC(C2(CC#C)CCC2)=O)C2CCCC1CC(NC(=O)Cc1c[nH]nc1O)C2 CCC(C)CC(=O)C(=O)NCC(C(=O)N1CC(C)(CSC)C1)N(C)C C1(C)(CNC(CN(CCC#C)C)=O)CC(F)(F)CN1C(c1ccc(Cl)s1)=O C1(C(N(CCC(C)NC(C(CC=CC)CC)=O)C)=O)CC2(CCOCC2)C1 C1(C(=O)NCC(CNC(C2CC(=C)C2)=O)OC)CC(CC)=NO1 C(=O)(C(F)CC(C)(C)NC(=O)CN1CCOCC1)N(CC(C)O)C1CC1 C1(NC(C2C(C#N)CC2)=O)CCOCC1C(=O)NC1CC(=C2CC2)C1 c1(CNC(c2n(CCCOC)nnn2)CCC2CC2)cccc2ccc(Cl)cc12 C#CC1(O)CCCN(C(=O)CC(CC=C)NC(=O)C(C)NC(=O)CC)C1 c1(C(N(CCN(C(CN2CCC(C)C2)=O)C)C)=O)cnn2c1OCC(O)C2 CCC(CN(C)C)C(=O)NC(CO)CCCNC(=O)C(C)(C)C C1(CC=C)(C(N2CCC(F)(CF)C2)=O)CCCN1C(c1cncnc1)=O c1(COC)ccc(C(=O)NC2CCC2NC(c2cc(C3CCC3)no2)=O)cc1F C1(CNC(C)Cc2cccc(Br)c2)CCOCCC1O C1(NC(c2cc(OCC)n[nH]2)=O)CCCN(C(c2scnc2COC)=O)CCC1 Cc1ncnc(C)c1CNC(=O)C(N1CCC(c2cccnn2)C1)=O C#Cc1ccc(C(=O)NC2(C)CCN(C(=O)Cc3ccc(Br)cc3)C2)nc1 CC1CN(C(c2ccc(C3CCOC3)cc2)=O)CC1NC(C1(C)CCOCC1)=O c1(C(=O)NCC(C)NC(=O)CCc2cncn2C)cc(O)ccc1N c1(C(=O)NCC=CCNC(C=CCN(C)CC)=O)cccc(-n2[nH]nnc2=N)c1 CCCCCCC(=O)NCC(C)(CC)NC(=O)Cc1ccc(O)c(F)c1 c1(OCCCNCCO)ccc(NC(C=CC(=O)NC(C2CCCO2)NC)=O)cc1 CCC(C(=O)N1CCC(NC(=O)CC2CNC(=O)O2)C1)N(C)Cc1ccccc1 C1(C(NOCC(=O)OC)=O)CC12CC(NC(=O)CN1CCC(C)C1)C2 CCCCCCCC(=O)N1CCC(CNC(C2CC(F)(F)CS2)=O)C(C)C1 c1(OC)cnc(C(=O)NCC(C2CC2)NC(=O)CCC(C)(F)F)c(OC)n1 c1(CNC(C(=O)N(Cc2n(C)ccc2)CC2CC2)=O)ccc(NS(C)(=O)=O)nc1 c1(C(=O)NCC(CC)NC(C2CC(=O)C2)=O)ccc([N+](=O)[O-])s1 N1(C(c2nncs2)=O)CCOC2(CCN(C(c3cncc4[nH]ccc34)=O)C2)C1 N1(C(Cc2nc(C)c(C)[nH]2)=O)CCCC(N(C)C(C2CCCCCC2)=O)CC1 C1(NC(=O)Cn2ncc(Br)n2)CN(C(C2CCOC2C2CC2)=O)CC1O n1(CC)nc(C(=O)NCC(F)CNC(c2c(C)n[nH]c2C)=O)ccc1=O c1(C(=O)NCCC(=C)CNC(C2COCCC2C)=O)coc2c(F)c(Cl)ccc12 C(=O)(C(C)CS(C)(=O)=O)N(CC(CO)(CO)NC(C(CC)OC)=O)C C1(C2CC2)(NC(=O)COc2ccsc2)CCN(C(=O)Cn2cnnc2)C1 CC(C)(C)CCC(F)C(=O)NCC1(O)CC(NC(C2(N(C)C)CCC2)=O)C1 CCCCCC(=O)NCC(=O)NCCCC(C)(C)NC(c1cncnc1C)=O N=C1NC(=O)C(CC(N2CCC(=CCNC(=O)CNc3ccncc3)CC2)=O)S1 c1(OC)c(C(=O)NC2CCN(C(=O)CCCC(C)(C)C)C2C)cc(Br)cc1F N1(C(CCNC(=O)OCC)=O)CCOC(C(C)NC(=O)CNc2cnn(C)c2)C1 c1(NC(C2N(C(CC3ON=C(C)C3)=O)CC(O)C2)=O)cc(C)cc(C)c1 N1(C(c2c(C(C)C)ocn2)=O)CCCC(O)(CNC(C2CCCC2(F)F)=O)CC1 c1(N2CCCC(COCC)C2)nc2ccccc2nc1NCCc1cccs1 C#Cc1cc(Br)ccc1NC(=O)C(=Cc1cc(F)cc(F)c1)C c1(C(N2CCCC(NCC)C2)=O)ccc([N+](=O)[O-])s1 c1(C(C(=O)NCC(CC)NC(c2cc(CN(C)C)c[nH]2)=O)(C)C)cccc(O)c1 C#Cc1ccc(C(=O)NCC2(F)CCCN(C(c3csnc3Cl)=O)C2)cc1C C(CNC(=O)C(O)C1CC1)(CCNC(c1ccc(C(C)=O)[nH]1)=O)OC C(=O)(C#CC1CCCCO1)NC1(OC)CCN(C(=O)CNC(C)=O)C1 C(CC(N)=O)(C(=O)N1CC(C#N)(CCF)C1)NC(C(CC1CCC1)OC)=O N1(c2nnn(C)n2)CCC2(COC(CNC(c3cccc4c3C(=O)NC4)=O)C2)C1 N1(C(C2(CC3CC3)CCC2)=O)CC2(CCC(C(=O)O)O2)C1.c1(C(=O)N)nnccc1SCC C(=O)(C(O)C(F)(F)F)N1CC(C(C)NC(c2cc(Cl)cnn2)=O)OCC1 C1(NC(C=C(C)C(C)C)=O)CC(N=c2nc(O)c3c(ncn3C)[nH]2)C12CCOCC2 N1(C(c2c(OCC)ccs2)=O)CCCN(C(=O)CC2CCCC23CC3)C(C)C1 c1(OCC(=C)C)ccccc1C(=O)NC(C)CNC(=O)Cc1cc(C)no1 C(C)(C)(CC(=O)NCC1(C)CCCN1C(=O)CCCc1nncn1C)N(C)C Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CC(C)N(C(=O)COCC(C)(C)C)C1 C(=O)(C1=CCCCCC1)NC(CC)C(=O)NOCC1(F)CCC1 C1(NC(C(CCC)OC)=O)CCCOC12CCN(C(c1nc(=O)n(C)[nH]1)=O)CC2 c1(C(=O)NCCSc2ccncc2-c2nc(CCCO)cs2)csc2ccccc12 CC1CN(C(=O)Cc2ccc(F)cn2)CCN1c1nnco1 CC1CN(C(C2CC2C(N)=O)=O)CC(C)N1C(C1CCCC1C1CC1)=O C1(C2CCN(C(=O)C(F)C(C)(F)F)CC2)(NC(CC(C)CC(C)(C)C)=O)CCC1 N1(c2ccc(C(=O)OC)cn2)N=C(C)CC(C)(C)CC1=O c1(-c2cc(CC(=O)Nc3c(NS(C)(=O)=O)cccc3)sc2)ccc(B(O)O)cc1 C(C)(N=c1nc(C(C)C)[nH]s1)c1ccc(CNC(C(C)Cc2ccco2)=O)cc1 c1(C(C(=O)NC(C(=O)OC)C)N(C)CC2CN(C)CCO2)cc(C)oc1C N1(C(C2(C(=O)NC)CC2C)=O)CC2(CCC(NC(=O)CN(C)CCOC)CC2)C1 C(=O)(C(C#N)C(C)C)NC(CC)(C)CNC(=O)CSc1cccc(F)c1 N1(C(c2cn(CCOC)nn2)=O)CC2CCCC(N(C)C(c3cnns3)=O)C2C1 c1(C(=O)NCC(CNC(C2CC(CC)C2)=O)O)oc2ccccc2c1COC C1(CNC(C(CC)OC2CCCC2)=O)(CNC(c2cnn[nH]2)=O)CCCCC1 c1ccc(C(c2nnnn2C2CC2)NCC2CC3CC3C2)cc1 CC#CCCC(=O)NCCC1CCCN(C(=O)CSc2ccc(OC)cc2)C1 C123C4CC1C1C(C4C21)C(C)NC3=O.c1(C(=O)NC(C)(C)CO)ccc2ocnc2c1 C1(OC)CC(CNC(=O)CNC(C)=O)N(C(c2cncc(C)n2)=O)C1 c1(CN(C2(C(F)F)CC2)CCN(C)C)ccc(F)nc1 C(=O)(C1CCCn2c(C)cnc21)N1C2C(NC(CNS(CC)(=O)=O)=O)(CCC2)CC1 C(=O)(C1=CCC2CCC1N2C(=O)CC1CC=CCN1C)N(CC(F)F)C(C)C c1(C(=O)NCC(CO)NC(CCc2ccc(C)s2)=O)cnn2c1CC(C)CC2 N1(C(C(C=C)(F)F)=O)CCC(F)(C(=O)NCc2cncc(O)c2)CC1 C1(NC(C2C(OC)C2)=O)CC2CC(NC(=O)COc3ccccc3F)CC2C1 c1(C(=O)NCCC2CCN(C(Cc3cn(C)nc3)=O)CC2)cc2occc2n1C C1(C(N(C(CC(=O)NC)C)C)=O)CCCN(C(=O)CCCSC2CC2)C1 N1(c2nc(Cl)nc(C)c2F)CC(CNC(=O)CCC(C)N(C)C)OC2(CCC2)C1 C12(C(=O)NCc3nc(CNC(=O)CC4CCCC4)sc3)CC3CC1C2C3O c1(NC(C)CCCCNC(C2(CF)CCC2)=O)ccc([N+](=O)[O-])c(O)n1 C(=O)(C1=CC2CCCC12)NC1(C)CCN(C(C23CC(CN2C2CC2)C3)=O)C1 n1(CC(N2C3C(NC(c4ccc(OC)nn4)=O)C(C3)C2)=O)nc2c(n1)CCCC2 c1(CC)ccc(C(N2CC(N(C)C(C3CC(CC4CC4)C3)=O)C(O)C2)=O)c(C)c1 C(CC(=O)N1CCC(C(=O)OC)O1)=CCNC(C(C=C)(C)CC)=O C#Cc1cc(C(=O)N(C)CC2CCCN(C(c3cccc(F)c3)=O)C2)cc(N)c1 C1(OC)CCN(C(C2(C)CCCN2C(c2cocn2)=O)=O)CC1 c1(NCc2c(F)cncc2-c2ccc(F)cc2)ncnc2ccccc12 C(=O)(C1=CCOCC1)N1CCC(n2cc(CN(C(CC(=C=C)C)=O)CC)nn2)C1 N1(C(c2ccc(C)nn2)=O)CCC2CN(C(=O)Cc3cc(C)ns3)CC2C1 C(=O)(CCC(=O)c1cc(C)sc1C)NCCCNC(C(C)NC(CC)=O)=O c1(C(=O)NCC=CCl)cc(CNC(C2CC3CC3C2)=O)no1 CC1=NOC2(C1)CC(C(=O)NC1CCCCN(C(c3cnn(C)n3)=O)C1)C2 N1(C(c2c(F)ccc(C#C)c2)=O)CCCN(C(=O)CCOCC2CC2)CC1CO c1(NC(C2C(C(N)=O)C2)=O)ccc(O)cc1.C12CCC(C1)C(=O)N2CC1CC1 CC(CC(F)F)C(=O)Nc1ccccc1SCCNC(CCCC#C)=O C1(CNC(CCN(CC)CC)=O)CCCCN(C(=O)CCC(C)NC(N)=O)C1 C1(CCC)CCCC1C(=O)NC(CC1CC1)C(=O)NCC1C2CCCC12 C(N=c1nc(N2Cc3c[nH]nc3C2)c2sccc2[nH]1)C1(C)CC(C)C1 C(=O)(C(C)(C)CC#N)N(CC(Cc1ccccc1)NC(COC)=O)C C1(C)(n2c(C(COC)OC)nc(-c3ccc(Cl)cc3)n2)CCS(=O)(=O)C1 c1(N(CCCOC)C)cc(=NCc2ccc(OC)c(Br)c2)cc[nH]1 N1(C(C2(NC(C)C)CC2)=O)CC(CNC(=O)CCOC2CC2)C2CCC12 c1(C(=O)NC2CC(NC(C3(N4CCOC4=O)CC3)=O)C2)cnc2n1CCOC2 N1(C(CCCNC(C)=O)=O)CCC2(CC1)COC(C(=O)NCCN(C)C)C2 Cc1nccc(CCC(N2CCC(CO)(NC(=O)COCC(C)(C)C)C2)=O)n1 c1(CCc2onc(-c3ccc(F)cc3)n2)nc2c(s1)CNC2 C(=O)(C(O)(C(F)(F)F)C1CC1)NCCN(C(c1n(C(C)C)ccn1)=O)C c1(OC)cccc(CC(=O)NC2CCCC2NC(c2cccs2)=O)c1.C1C(=O)O1 CN1CCN(C(c2ccc(Cl)o2)=O)C(CN2CC(CO)(Cc3ccccc3)C2)C1 C1(C(=O)NC(CNC(c2c(N)sc3c2CCC3)=O)CO)Cc2cc(F)cc(F)c2O1 C1(C(=O)NC(COC)CNC(c2cnc(SC)s2)=O)CCCSC1C c1(OC)cc(C(N2CC(CNC(C3(C)CC3F)=O)C2)=O)cc(F)c1F O=C1NC2CN(C(=O)CC3CC(NC(c4cc(O)no4)=O)C3)CC2N1 N1(C(C(C)(C)N(C)C(c2cn(C3CC3)nn2)=O)=O)CCCC(C(C)(C)C#N)C1 N12CC(C(C)(C)C1)NC(=O)c1cnc2cn1.c1(C(=O)OC)cnc(SC)o1 C(=O)(C(C(C)NC(=O)CC1CCOC1(C)C)C(C)C)NC(C(=O)N(CC)CC)C N1(C(C(c2cccc(OC)c2)O)=O)CCN(C(C2(C)COC(=O)C2)=O)CC(O)C1 c1(NC)cncc(C(=O)NC(C)C=CC(=O)N(C(C(N)=O)C2CC2)C)c1 c1(CNC2CC3CN(C(=O)OC(C)(C)C)C2C3)ccc2c(c1)C(=O)NCC2 c1(NC)cnc(CNC(C2CC(n3cccn3)C2)=O)cn1 C(=O)(C#CC1CCC1)NCCCCN(C(c1c(CC)noc1C)=O)C c1(C(=O)NCC(CC=C)NC(c2csc(CO)n2)=O)cnc(Cl)c(C2CC2)c1 N1(C(c2cc(CC)oc2C)=O)CC2(C)CN(C(=O)Cc3csc(C)n3)CC2(C)C1 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC1CN(C(C2CC(C)CC(C)C2)=O)C1 c1(C(=O)NCCCC(C)NC(c2cc(O)no2)=O)cc(Cl)cc(Cl)c1 c1(CC)cc(N2CCCC(C(=O)NC(c3ccnn3C)C)C2)ncn1 C=C(CNC(=O)C1=CCC(NC(C2CCC(C)(C)CC2)=O)C1)c1ccccc1 c1(C(=O)NCc2cc(C(=O)NC3CC(COC)C3)sc2)cccc(=O)o1 c1(C(N2CC(N(C(CCC#C)=O)C)C(C)CC2)=O)cc[nH]c2nccc1-2 N1(C(C(C)CN2CCOCC2)=O)CC=C(CNC(c2cc(F)cc(Cl)c2)=O)CC1 CN1CCC(C(=O)NCCSC2CC2)(NC(=O)C(C2CCOCC2)=O)C1 C12(CC)CN(C(=O)C=C(C)C(F)F)C(CNC(=O)CC(C)c3ccco3)(C1)C2 c1(C(N2CCC(C(C(=O)N(C(CC)C)C)F)C2)=O)noc(CC)c1C N1(C(CCOCCN(C)C)=O)CCOC2(CCN(C(C3CCC3(F)F)=O)C2)C1 C(=O)(C(C)COC(c1ccccc1)=O)NCC(CNC(CNC(=O)NC)=O)C C=C(C)C(CC(=O)N1CCC(C(N2CC(C3CCCOCC3)C2)=O)CC1)OCC C12(C(=O)NCC3(NC(=O)C4CC4)CCC3)OCCCC1C2(F)F.c1ccccc1Cl c1(C(=O)NC2(C)CN(C(C(CC)c3ccccc3)=O)C2)c[nH]c(=N)cc1C c1(C(=O)NC2C(CNC(=O)CCC3NC(=O)NC3=O)CC2)cc(F)c(F)cc1O C1(CNC(C(COC)(C)C)=O)CN(C(c2ccc(C3CC3)s2)=O)CC(C)(C)C1 CCC(C)(C)C(O)C(=O)N1CCC(C2(NC(=O)C=Cc3cccc(O)c3)CC2)C1 N1(C(C(=O)NCC=C)=O)CCN(C(=O)CCn2ccnn2)CC1.C(=O)(COC)NCC C1(NC(c2c(C)nns2)=O)CN(C(=O)C(C2CCCCC2)O)CC1n1ccnn1 Cc1cccc2c(C(=O)NC3CCN(C(C45CC(F)(CO4)C5)=O)C3)coc12 C(=O)(C1=CCCC1C)NCC(CC)NC(=O)CCc1ccc(F)c(F)c1 C(CC)(C(=O)NCCC1CC(NC(c2cc(C)on2)=O)C1)OCC C1(NC(c2cc(OC)ncc2)=O)(CO)CCCN(C(C2CC3(CSC3)C2)=O)C1 CC(CCCCNC(C1(CO)CCOCC1)=O)NC(=O)C(C)SC(F)(F)F N1(C(CCC(=O)C(F)F)=O)CCCCCCC1C(=O)NCCN(CCO)C1CC1 c1(C(N(C)CC2CCN(C(c3csc(CO)n3)=O)CC2)=O)cccc(Cl)c1F N1(C(c2c(CC)con2)=O)CC(NC(C23CCC(CO)(CC2)C3)=O)CC(C)C1 c1(CC(C)C)n[nH]c(=NC2CC3CN(C(C4CCC(N=[N+]=[N-])CC4)=O)CC23)s1 c1(C(C)NC(CCn2cc(-c3c(C)noc3)nn2)=O)ccc(OC(F)F)cc1 C=CCC(CC)C(=O)N1Cc2ncsc2C1.c12ocnc1C(=O)OC2 c1(OC)c(C(=O)NC2CCC(N(C(=O)C(O)C3CC3)C)CC2)ccnc1F N1(C(CS(CCC)(=O)=O)=O)CCC2(CC1)CC(N(C(c1cc(C)sn1)=O)CC)C2 C1(C(=O)NC(c2noc(C3CC3)n2)(C)C)CCN(C(c2ccsc2)=O)C1 CN=c1cc(C(N2CCOC(CN(C)C(C3CC4(CSC4)C3)=O)C2)=O)cc[nH]1 CC1(C)CCCC(C(=O)NC2CCCC2NC(C2(c3ccccc3)CC(O)C2)=O)C1 CC1(C(=O)NCC2CCCCN(C(C3CCS(=O)(=O)N3)=O)C2)CCCC1(F)F C(c1c(F)cccc1F)=CC(=O)NC12CN(C(C(C)NC(C3CCC3)=O)=O)C(C1)C2 N1(C(c2ccc(C)n2C)=O)CC(C2CC2)(C(N2CCC(F)C2)=O)C1 Cc1ccc(C=CC(=O)N(CCC(C)NC(=O)COc2ccccc2C)C(C)C)s1 Cn1nc(C(N2CC3CC(C2)C3NC(C2CCCO2)=O)=O)c2c1CCCC2 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NCCN(C(CC=C=C)=O)CCOCCO c1(CC(=O)NC2C3(CN(C(CN4CC(C)C4)=O)C3)CC2)ccc2c(c1)NC(=O)C2 N1(C(CC=C)=O)CCCC2(CCN(C(C3CC4CC3C4)=O)C2)C1 c1(N(C(C)C)C)ccc(C(=O)NC(C)CCCNC(C2COC(=O)C2)=O)cc1 N1(C(C2CCCC2O)=O)CC2CCN(C(=O)CCCc3ccncc3)CC12 C1(CO)CN(Cc2cc(CNC3CCC3)ccn2)CC12CCC2 CCCCS(=O)(=O)NC(C)C(=O)N(C)CC1CCCN1C(=O)CC1OCCO1 N1(C(C)=O)CCN(C(=O)CCn2cc(-c3cnc(C)o3)nn2)C(C)C1 c1(C(C(=O)NC2CCC2)N(CCCCOC)C)ccc(OC)c(Br)c1 C1(C(N(CCC(=O)N(C)C)C(C)C)=O)CCCCN1C(=O)CCC1CCCCO1 S(=O)(=O)(c1ccc(NC(C2CCC3COCCC3NC2)=O)c(C(=O)O)c1)N(C)C c1(C(N2CCCC(NC(C(=O)NCC)=O)C2)=O)cccc2sc(C(F)(F)F)nc12 CC(C)C(CC(=O)N1Cc2ncsc2C1)NC(C1CCC2(CCC2)C1)=O C12(C(=O)NC3C(CNC(CCc4[nH]c(=N)sc4)=O)CCCC3)CC(C1)S(=O)(=O)C2 CCCC(C(=O)N1C(C(=O)NCCCC(C)(F)F)CCC1C1CC1)OC c1(COCC)ccc(C(=O)NC(C)C)cc1.C12CC1C(=O)N2.C(=O)(CO)N c1(Nc2ccc3cnc(C)n3c2)[nH]c(=N)nc2c1ncn2CCO OCC(F)(F)C(c1ccccc1)NC(=O)C(c1ccc(Cl)cc1)C1CCC1 c1(CC(N2CC3C(CNC(=O)Cc4cccs4)(C3)C2)=O)ccc(O)c(Cl)c1 c1(C(N(CCCNC(C(CC)OCC)=O)C2CC2)=O)ccc(N(C)C)cc1.C(C)(=O)N c1(C(=O)OC)cc(S(=O)(=O)N2CC3(CCC(NC(=O)CO)C3)C2)ccc1C N1(C(CCCOCC=C)=O)CCCC(CNC(=O)C=CI)C1 Cn1ccc(=O)c(C(=O)NCC2CCCC(NC(c3ccc(Cl)[nH]3)=O)C2)c1 c1(NC(CNC(C(C)NC(c2csc(C(F)(F)F)n2)=O)=O)=O)ccc(C(F)F)nc1 c1(C(N(C2CN(C(C3C(OCC)C3C)=O)C2)C)=O)ccn2c(C)cc(C)nc12 N1(C(C(C)CC(F)F)=O)CCC2CN(C(=O)CC3CN4CCC3CC4)CCC2C1 N1(C(C(=O)NC2CCC=CCC2)=O)CCC2(CCCO2)C1 c1(CC(=O)NC(C)CNC(=O)CC2CCN(C)C2=O)cc(F)ccc1Br CC(C)(O)C(F)(F)CNC(c1ccc(CNC(c2nsnc2O)=O)o1)=O Cc1cc(C)c(C(N2CC3CC(NC(=O)CCC4CC4(C)C)C2C3)=O)c(C)n1 N#Cc1cc(F)c(C(N2CCCC3(C2)CN(C(C2(F)CC=CC2)=O)C3)=O)c(F)c1 c1(C(N2CC(NC(c3[nH]cc(C)c3)=O)C(F)C2)=O)ccc(C2=CCOCC2)cc1 N1(C(CC)=O)CCC(CNC(c2cc3c(Cl)cccn3n2)=O)C(F)(F)CC1 C(=O)(C1SCCc2ccccc21)NC1CC(NC(COCCCC)=O)C1 N1(C(=O)Nc2ccc(Cl)cc2)CC2CCN(c3nccc(OC)n3)CC2C1 Cc1ccc2c(c1)CN(C(=O)CN(C(C1CCC(C(N)=O)C1)=O)C(C)C)C2 c1(OC)cc(C(N2CC(NC(c3cnc(O)cc3C)=O)C3CC23)=O)ccc1C c1(OC)c(C(N2CC3CC2CN(C(c2cnc(SC)s2)=O)C3)=O)nc(O)nc1O C1(C(N2CC(CNC(=O)CCCNC(=O)CC3CC3)C2)=O)CCC(F)(F)CC1 C#Cc1cc(F)c(C(=O)NC23CCC(NC(c4nnc(C)s4)=O)(CC2)C3)cc1F N1(C(C(CC)(C)O)=O)CC2CC1CC2NC(c1cccc(C)c1)=O c1(OC)ccc2c(CN3CCC(NC(C4C5COCC45)=O)C3)cc(=O)oc2c1 C1(NC(c2cc(C(C)C)no2)=O)CC2(C1)CC(NC(=O)C=CC(F)(F)F)C2 c1(C(=O)NCCCN(C(c2c(C)nc[nH]2)=O)CCO)ccc(-c2ccco2)nc1 N1(C(=O)C2=COCCO2)CCC(C2CCN(C(c3c[nH]nc3C(F)F)=O)C2)C1 C(=O)(C(C)(O)CCN(C)C)N1CC(CN(C(C2ON=C(CC)C2)=O)C)OCC1 N1(C(C(C)NC(C2(CC)CCOC2)=O)=O)CCC(F)(COC)CC1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCC(N(C)C(C2(C#N)CC3(CC3)C2)=O)C1 C(=O)(C(C)CC(F)(F)F)NC(c1ccccc1)CNC(c1c(CC)c[nH]c1)=O c1(CN(C(N2CC(CC)N(C3CC3)CC2)=O)CC)cc([N+](=O)[O-])cn1C C1(C(=O)NC23CN(C(CSC(C)C)=O)C(CC2)C3)COc2ccc(Cl)cc2C1 C1(CNC(C(CC)(C)O)=O)CC2(CC2)CN1C(=O)Cn1ncnn1 C(=O)(C(C)(O)CC)NCC(CNC(C(CC)C1CCC(=O)N1)=O)C N1(C(C(=O)NCCOC)CC2CCCOCC2)CCc2ccccc2CC1 Cc1[nH]nc2c(-c3cc(C(=O)NCC4CCCO4)c4n[nH]cc4c3)cccc12 N1(C(C(c2ccc(F)cc2)OC)=O)CCN(C(=O)CCC2CC2)CC1CCOC CC1CN(C(C2CCC2)=O)C(C)CN1C(c1ccccc1C#N)=O c1(CC(C)C(=O)NC2CCN(CC(=O)NCC3CC3)CC2)ccccc1F n1(COC)nccc1C(=O)NCC1CCCC1NC(=O)C(=O)NC(C)C C1(C(=O)NC2CCN(C(C3(OC)CCCC3)=O)CC2O)CCc2n[nH]cc2C1C Cc1csc2c(C(=O)N(C(C)CNC(c3coc(S(N)(=O)=O)c3)=O)C)ncnc12 c1(C(N2CCN(C(=O)C=Cc3cnc[nH]3)C(C(F)F)C2)=O)nnn2c1CSCC2 N1(C(CSCCC)=O)CCN(C(C2(C)C=CCC2)=O)CC2(CC2)C1 Cc1ncc([N+](=O)[O-])cc1C(=O)NC(C(C)NC(C1(CC(F)F)CC1)=O)C(C)C C1(N(C(c2nc(C)sc2)=O)C)CC2CC1N(C(C13CC4CC1C3C4O)=O)C2 CCCC(C(=O)NCC(C)NC(=O)C(F)=C1CCCC1)c1ccccc1 c1(OC)ccccc1CCC(=O)NC1(CNC(=O)Cc2ccccc2)CCC1 C1(CCNC(C(C)(C)Cl)=O)CCN(C(c2ccnc(C3CC3)c2)=O)CC1(F)F N1(C(C(C(C)O)C)=O)CCN(C(c2ccccc2Br)=O)C(CO)C1 C(C(=O)NCCCCCCN(C(=O)CSC(F)F)C)(C(C)C)OC C(=O)(C#CC1CCOCC1)N(C)CCNC(C1CCC1)=O c1(OC)cc(C(N2CCOCC2C(=O)NCc2cccc(Cl)c2F)=O)ccc1Cl c1(N(CC(C2CCCOC2)O)C)cccc(-c2nn[nH]n2)c1 N1(C(C2(C#N)CCCO2)=O)CC(CNC(c2csc(S)n2)=O)C2(CC2)C1 C1(C(=O)NCc2cnc(C)o2)CN(C(=O)C(=O)C(C)C)CC12CC2 Cc1cc(N)n2ncc(C(N3CCCC(C(=O)NC(C)CO)C3)=O)c2n1 c1(C(C)NC(=O)CCC(F)(F)Br)ccc2c(c1)CCCC2=O C1(NC(CCCC)=O)CCC(N(C(=O)CCC2CC2(F)F)C)CC1 c1(C(=O)NC(CC(=O)O)C(F)(F)F)cnc2c(c1)OCO2 N1(C(CCCOC(C)C)=O)CC(CNC(=O)CCC(N)=O)N2CCC1C2 N1(C(=O)CCc2ncc[nH]2)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1 c1(C(N2C(CN(C(C(CC3CCCCC3)OC)=O)C)CCC2)=O)ccc(Cl)cc1 C(=O)(CCCC(C)=O)NC(C1(O)CCN(C(CC2(OC)CCC2)=O)C1)C N1(C(c2nn(C)cc2I)c2n(C)nnn2)CCOC2(CCSC2)CC1 N1(C(C2CCC(C)CC2)=O)CCCN(C(C2(F)CCC2)=O)CC1 N12CC(C3CN(C3)C(=O)c3cn(CC)c(n3)CC1=O)C2.C1(COCC)(CC)CC1 N1(C(c2ccc(O)nc2Cl)=O)CC(CO)C2(C1)CN(C(C13CSCC1C3)=O)C2 c1(C(N2CCCCCC(NC(=O)Cc3ccon3)C2)=O)cccc2c1CCO2 N1(C(c2nc(C)oc2C)=O)C2CCC(C2)C1C(N1CCC(n2ccnc2)C1)=O Cc1nc(C2CC2)ccc1-c1nc(N(C)C)n[nH]1 N1(C(C(C)OC)=O)CCC2(CCCN2C(C2CCC(=O)NC2)=O)C1 C(CN=c1[nH]c(Cl)ncc1C(=O)OC)OC(c1c(OCC)ccc(C)c1)=O CCC(CC(=O)NC1CCCC1CNC(=O)C(C)CN(C)C)c1ccccc1 C1(C)(CNC(c2c(CC)n[nH]c2)=O)CCCN(C(=O)CCNC(=O)COC)C1 N1(C(CC2C(C)(C)CCCO2)=O)CC2CCC(C1)N2C(=O)C1=CCSC1 CC(=O)CCCCC(=O)NC(CO)C(=O)N(CC1=CCCOC1)C Cc1cn2c(C(=O)NC3CN(C(=O)CSc4nc[nH]n4)CC3C(F)F)cnc2s1 C1(NCc2n(C)nc(C)c2Br)CCCC(C)C1C C1(CNC(C2C(c3n(C)cnc3)C2)=O)C(O)C(O)CN1C(=O)CC1=CCCC1 C(=O)(CC(C)(C)CC(F)(F)F)NC1(C)CCC(NC(c2cn(CC)nc2)=O)CC1 CCCCCCCC(=O)N1CC=C(CCNC(C2(CO)CC2)=O)CC1 CC1CN(C(c2cccc(-c3ccsc3)c2)=O)CCN1C(c1cccs1)=O CC(C)C(CCC(=O)NC1CCC(=O)NC1)NC(c1cnc[nH]c1=N)=O c1(C(N2CCCCC(C)C2)C(=O)NCCC2CC2)nc2ccccc2s1 c1(C(N2CCC(CNC(C3CC34CCCOC4)=O)CC2)=O)cccc(F)c1F C1(CC(C)C)(C(N2CCC(N(C)C(c3nnn(C)c3N)=O)C2)=O)CCNC1=O N#Cc1ccc(C(N2CC(F)CC2C(=O)NCc2cncs2)=O)cc1F c1(C(=O)NC(C(C)NC(c2n(CC)c(O)nc2)=O)C)ccc2c(c1)OC(C)(C)C2 C1(NC(C2C(c3c(C)cccc3)C2)=O)CC(C)CN(C(=O)CSC(F)F)C1 N1(C(CCC(N)=O)=O)CCC(O)(CNC(c2n[nH]c3c2CCC3)=O)CC1 CCC(CNC(C1CN(C(C2CCC2COC)=O)CC1C(C)C)=O)CC(C)C C#Cc1cc(C(=O)NC(C)(C)C(C)NC(C2COCCO2)=O)ccc1C C(C)(C)(C(F)(F)F)NC(CCC1N(C(c2c(C)nsc2)=O)CCC1)=O N1(C(CCOCCC)=O)CCOC(CC(=O)NC(C2CCOC2)CO)C1 c1(C(N(C2CCN(C(=O)C(F)F)C2)C)=O)cnc2ncnn2c1O C(=O)(C(C)(C)CCO)NC1CCC(Cn2cc(-c3c(C)c[nH]n3)nn2)CC1 C1(OC)CC2(C1)CC2C(=O)NCC(O)CNC(=O)CCc1ccccc1F c1(C(=O)NCCC)ccc(O)cc1.C1(C(=O)Nc2cc(CO)cs2)CCC12CCC2 c1(OC)cc(F)c(C(=O)NCC(C(C)C)NC(c2cc(C)cnc2N)=O)c(F)c1 N1(C(CCC=C)=O)CCCC2(CCCN(C(c3cc(C(F)F)no3)=O)C2)C1 CN1C(=O)C(F)CC1C(=O)NCC1(NC(c2sccc2OC(F)F)=O)CCC1 c1(C(=O)NCCOCCN(C(Cc2ccn(C)n2)=O)C)ccnc2ccsc12 C1(C(N2CC(CCCCNC(CCc3cc(C)no3)=O)C2)=O)CCOC(=O)CC1 S(=O)(=O)(c1ccc(NCC(C)(C)CC(F)(F)F)nc1)NC(CCC)CO c1(CCC(=O)NCCC2N(C(C(C)OC)=O)CCC2)ccncc1Br c1(NC)cnccc1C(=O)NCC(C)CNCC1COCCN1C(=O)CC1CC1 C1(CCC(=O)NCC(CC)C#N)CCCCN(C(C2CC(F)CN2C)=O)C1 c1(C(C)NC(=O)NCC2N(CCC)CCC2)ccc(Br)cc1Cl C1(CC(=O)NC(C(C)C)CNC(C2CC3(C2)CC3F)=O)CCCCC1(C)C N#Cc1ccc(C(N2CCCC(O)(CNC(c3ccccc3Cl)=O)C2)=O)cc1F N1(C(C(C)C2CCOC2)C(=O)NC2CC2)CCCC2(CC1)CNC(=O)O2 C(=O)(C(F)CC1CCC1)N(C1CCCCC1)C(CN(C)C(c1ccsc1Br)=O)(C)C c1(-n2cc(C(C)NCC(F)(F)F)nn2)ccc(OCCN2CCCCC2)cc1 N1(C(CN(C)S(N)(=O)=O)=O)CCc2[nH]nc(CNC(C3(C)CNC(=O)C3)=O)c2C1 N1(C(C2CCC(n3cc(C(CC)O)nn3)C2)=O)CCC(S(=O)(=O)C2COC2)CC1 C1(N(C(CN(CC(C)F)C2CC2)=O)C)CCCC1C CCC(CC)C(F)C(=O)N1CCCC1C(N1CCCC(N2CCCC2)CC1)=O CC1CN(C(=O)Cc2cccc(Cl)c2F)CCN1C(c1cc(F)ccc1F)=O c1(-n2ccc(CN(C(c3cc(CC)[nH]n3)=O)C3CC3)n2)ccccc1C CC1OC(C)C(Cn2cc(CN3CC(Cc4ccccc4)C3)nn2)C1C N1(C(CCC2COC(C)(C)O2)=O)CCC2(C1)CN(C(C1(C)CCC(=O)NC1)=O)C2 C(C(C(C)(C)C)NC(c1cncc(F)n1)=O)NC(C(C1CCOCC1)C)=O N1(C(c2n(C)c3c(c2)occ3)=O)CCC2(C)CN(C(c3cc(Cl)n[nH]3)=O)CC12 C(=O)(C1=COCCO1)NCC(CC)(CC)NC(c1ccc(Cl)c(C(F)(F)F)c1)=O C1(CC(=O)N(CCN(C(C(CC)SC)=O)C)C(C)C)CC2(CCCC2)CO1 C1(CNC(C(C)CC2CCCO2)=O)CCC(NC(c2cc[nH]c2)=O)CC1 c1(C(N(CCNC(=O)COc2cccc(Br)c2)C2CC2)=O)cc(O)nc(O)n1 N1(C(CNC(CC)=O)=O)CC(CNC(C2(c3cc[nH]n3)CC2)=O)C(C)C1 C(C(C)C(=O)N(C)CCN(C(=O)CC1(C(F)(F)F)CC1)C)OCC C1(C(=O)NC(COCC)C(C)C)CC(CC)CCN1C(c1ccnc(O)c1)=O c1(C(C)C(N2CC(c3cccc(F)c3)C(O)C2)=O)ccc(C#N)cc1 Cc1ccc(-n2nc(CC3COC3)nc2Cn2cc(Br)cn2)cc1Cl c1(C(=O)NCC(CC)NC(C2CCCC2(F)F)=O)c(C(F)F)nc2ccccn12 c1(CNC(C2C(C#N)C2)=O)ccc2c(c1)CCCC2NC(c1ccc(F)cc1)=O C(=O)(C(C(C)(F)F)NC(=O)CCc1ccccc1C(F)(F)F)OCC C1(NC(CCCSC)c2nnnn2CCC2(C)CC2)CCOC2(CCOCC2)C1 c1(CC(=O)N(CC(C)NC(c2cncc(CC)c2)=O)C)ccc(C)c(O)c1 N(C1CC(C)n2ccnc21)C(C(CNC(c1ccn(CC)n1)=O)(C)C)=O CC1(C)CCC(C)(NC(=O)C(NC2=COC(C(C)(C)C)NC2)=O)CC1 O=S(=O)(c1[nH]c(=NCC2CCCO2)ccc1Br)N1CCCC(OCC2CC2)C1 C1(CCC)CCCN1N1CC(C)(C)OC(CC)C(CC)C1 C(=O)(C(C)CCCC(C)=O)NC(CCC(=O)NC(C(=O)OC)C1CCC1)C(C)C C(=O)(C(O)CCc1ccccc1)NC(CNC(c1nc[nH]c1CO)=O)C1CCC1 C1(C(=O)NCCN(C(=O)CC2CCCC(=O)C2)CC)CC2OC1C1CC21 C1(C2CCN(C(=O)CC3(C(F)(F)F)CC3)CC2)(NC(c2cccs2)=O)CCC1 Cc1c(C(=O)NC(C)(C)CNC(=O)C(C)O)[nH]c2c(C)cccc12 N1(C(C=C(CC)C)=O)CCOCC1CN(C(=O)C(C)(C)Cc1ccccc1)C C1(C(=O)NC2CCN(C(Cc3c(C)nc(SCC)s3)=O)C2)CC(=O)OC1(C)C N1(C(CCCCNC(c2csc(C)c2C)=O)=O)CC(CO)C2(CCC2)C1 C12(NC(=O)COC3CCCCC3)CCCC1N(C(=O)CCc1ccco1)CCC2 N1(C(C(=O)N(C)C)=O)CCC(NC(C2(C)CCN(C)C2=O)=O)C(CO)C1 N1(C(C(C2CCC2)OCC)=O)CCC2CCCC12C(=O)NC1CC12CCCCC2 Cc1ccc(C(=O)NC2CCOCC2NC(=O)C(C)(F)F)c2ncccc12 CC1CC(NC(c2cc(C(C)(C)C)on2)=O)CN(C(c2cccn(C)c2=O)=O)C1 c1(N2C3CC(=O)NCC2CC3)nc(NC2COC3(CCC3)C2)c2ccccc2n1 N1(C(c2cccc(C)c2)=O)CCC2(CCCN(C(c3ccnn3C(C)C)=O)C2)C1 CC1CCC(NC(C23CCN(CC2)C3)=O)CN1C(C1CCN(CC(F)F)CC1)=O c1(C(=O)NC(C2CCN(C(C3C(C)C3C)=O)C2)C)cn(C2CC2)cn1 CC1CCN(C(c2cccc(-c3ccccc3N)c2)=O)CC1(F)F CCS(=O)(=O)c1ccccc1CN(C(=O)C(N)=O)C Cc1cc2c(C(=O)NC(CNC(C3CC(C)(C)CO3)=O)C3CC3)ccc(C)c2[nH]1 C1(OC)(CNC(c2cnc(CC(C)C)s2)=O)CN(C(C2CCCN2C(C)C)=O)C1 C(=O)(CCCC(=O)N(CCN(C)Cc1ccnc(Br)c1N)C(C)C)OC c1(C(N2CC(CCNC(C3(OC)CS(=O)(=O)C3)=O)OCC2)=O)cc(C)ncc1C C1(c2nc(=N)[nH][nH]2)CCN(C2CCCCC2)CC1 C(=O)(CS(=O)(=O)C(C)C)NCC(C1CCN(C(C(C(C)C)(C)O)=O)CC1)C c1(C(=O)OCC)cccc(CC(=O)NCCO)n1.C12CC1CC2=O.C1(O)CCC1.CC C1(CNC(=O)NCCC(CC)(F)F)CC(OC)C12CCC2 N1(C(c2nc(C)nn2C)=O)CCC(CO)(CNC(C2C3CCCCCC23)=O)CC1 CC(CNC(=O)CC(=O)NCCN(C)C)C(=O)NCCO C(=O)(C#CC1(C)CCCO1)N1CC2N(C(CCC3CCCN(C)C3)=O)C(C2)C1 C1(O)(CNC(C2CC(NS(C)(=O)=O)C2)=O)CCCN(C(C2CC23CCC3)=O)C1 Cc1cc(C(N2CCCCC2CN(C(=O)CCC2CCC(=O)NC2)C)=O)n(C)n1 C1(CNC(c2c(CC)onc2C)=O)CC2(CC2)CN1C(c1cccc(NC)n1)=O C1(C(=O)NC(C(CO)NC(c2c(C)nn[nH]2)=O)C)Cc2cc(Br)ccc2O1 CC1(C)CC(c2ccc(F)cc2)(C(=O)N(CCNC(C2CC2C#N)=O)C2CC2)C1 CC(CNC(=O)CCNC(c1ccc[nH]1)=O)CN(C(=O)COc1ccsn1)C C1(CNC(c2c(C)cc(C)s2)=O)CCC(C)(C)CN1C(c1ccc(=N)[nH]c1)=O c1(CCC(=O)NC(CC)(C)CNC(c2csnc2C)=O)cccc(F)c1 C(=O)(CC(C)CC(C)C)N1CCN(C(C2(OCC)CCCC2)=O)CC1CF C1(C)(CC)CCC(C(N2CC(CF)(NC(c3ccnn3CCOC)=O)C2)=O)O1 C1(C(=O)NC2CN(C(c3c(C)nc[nH]3)=O)CC(F)C2)CCc2ncccc2C1 Cc1c[nH]nc1C1(C(=O)NCCN(C(=O)CC2CC=CCC2)CC2CC2)CC1 C(=O)(C(C)(C)CC(C)=O)NCC(CNC(C(CC)SC)=O)(C)C O(N=C1CCCCC1)CC(=O)NCC(C)CNC(=O)CC1CCCSC1 c1(CN=C(NC(C)C)NC(C)(C)CF)ccc(F)c(F)c1 N1(C(C2C(C)(CC)C2)=O)CCOC2(C1)CN(C(c1c[nH]c3nccc-3c1)=O)C2 C(=O)(CCCCCCNC(=O)CC1CCCO1)NCC(CC)CC N1(C=O)C2C=C(c3ccccc3)CC1CC2.CC1COCCC1NCCN(C)C CCC(C)(CNC(=O)C(C)Cn1cccn1)NC(=O)CNC(c1ccccc1)=O C1(NC(CCn2ncc(C)c2)=O)(CO)CCCN(C(C2CC(F)(CO)C2)=O)C1 N1(C(C2(SC)CN(C(=O)C(C)C3CCOC3)C2)=O)CCC(=O)N(C)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CCC2(C)CN(C(=O)COCC(F)F)CC12 CC1CN(C(C2CS(=O)(=O)C2)=O)CC1NC(=O)CSc1nncn1C1CC1 C1(C(=O)NCC(C)(C)OCC(=O)N(C(c2onc(C)n2)C)C)CC(=O)NC(C)C1 C(=O)(C1=C(C)C(C)(C)OC1=O)NCCCC(C)NC(CC(CC)O)=O c1(SC)ccc(C(N2CCSC(C(=O)Nc3nc(O)cs3)C2)=O)c(C)c1 c1(CC(N2CC(C(=O)OC(=O)N(C)CC)C2)=O)ccc(-n2c(C)ccc2C)cc1 C1(CNC(C(C2(C)CC2)NC(C(=Cc2ccco2)C)=O)=O)CN(CC)C(=O)O1 C1(N(C(C(CSC)O)=O)C)CCCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 c1(NCC2OCC(CNC(c3cc(CC)n(CCO)n3)=O)C2)nnc(C)c(C)n1 c1(C(=O)NCC(CC=C)NC(c2ccc(F)cc2O)=O)ccn2cnnc2c1 C1(NC(C(C(C)O)NC(N)=O)=O)CN(C(=O)C(=O)N=S(C)(C)=O)CC2(CCC2)C1 n1(CCC)cccc1C(c1nnnn1CC1CCCO1)NC1(CC2CC2)CC1 C(=O)(C(C)(F)C(C)(C)F)NCC1(NC(c2c(C)scn2)=O)CCCCCC1 C1(CNC(C2(CC)COC2)=O)C2CN(C(=O)C=Cc3ccc(C)o3)CC12 c1(C(N2CCC(=CC(=O)NCc3cccc(O)c3)CC2)=O)ccc(Br)cc1F c1(C(=O)NCC2CN(C(C(C(CC)C)N(C)C)=O)C2)c(OC)ccc2c1CCC2 N1(C(C2(COC)CC2)=O)CC2CC(O)C1C2NC(c1cc(C(C)(C)C)[nH]c1C)=O C1(C(=O)NCCc2ncc(C)cn2)N(C(C2C3CCCOC23)=O)CC12CCCC2 c1(SCC(=O)NCC(C)(C2CCC2)NC(CCSCC)=O)ccccc1C c1(C(C2CCC2)OC)nc(C2CC23CC3)nn1-c1ccc(Cl)nc1 N1(C(C2(COC)CC2)=O)CC=C(CC(=O)NCCC2(C)CCOCC2)CC1 N1(C(CNC(CNC(C)=O)=O)=O)CC(CNC(=O)C(C)(C)CO)CC12CCC2 C1(SCCOCCNC(C2C(C(N(CC#C)C)=O)C2)=O)CC(=O)N(C(C)(C)C)C1 C1(C(=O)OC)CCC(NC(C2CC2C2CC(F)(F)C2)=O)C(C)C1 c1(C(C)=O)ccc(C(N2CCCC(CNC(C3(O)CCC3)=O)CC2)=O)cc1C Cc1ccoc1C(N1CCC(C(C)C(N2CCOCC2)=O)C1)=O C(CCN(C)C(c1cccnc1O)=O)(C(C)C)NC(C1(CC)CCCC1)=O C12(C(N3CCOCC3)=O)CCOC(CNC(c3cc(CCC)c(C)s3)=O)(C1)C2 N1(C(c2cnc(CC)s2)=O)CC2(COC(CNC(=O)C3=CCCOCC3)C2)C1 N1(C(C#CC(C)C)=O)CCC(C)(C)CC1C(=O)NCC(C)(O)CC(C)C Cc1cc(C)c2c(c1)CCC2NC1CCCC(N)CC1 CS(=N)(=O)C1CC12CN(C(C1CCCCN1C(=O)CC1CSCCO1)=O)C2 C=CC1CCN(CC2CCC(C(=O)O)CO2)CC1 C1(C)(CNC(CCC=C=C)=O)CN(C(C2(CS(N)(=O)=O)COC2)=O)CCO1 N1(C(c2n(CC)nc(C)c2)=O)CCC(C)C(NC(=O)CCc2cnccn2)C1 CCCC(C)CC(C(=O)NC1CC(C(=O)OC)C1)N1CC(CC)C(CC)C1 N1(C(C)=O)CCN(C(C2CCN(C(c3cc4sccc4s3)=O)C2)=O)CC1(C)C C1(CC)(NC(C2CC=CCC2)=O)CCCN(C(=O)C(C2CCCN(C)C2)(C)C)C1 c1(C(=O)NC2CCN(C(C#CC3(CC)COC3)=O)C2)cc2c(cc1N)OCCO2 C(=O)(C1Cc2ccccc21)N1C(C(=O)NOCc2cccnc2)CCCCC1 N1(C(C)=O)CCN(C(C2CCC(O)CN2C)=O)C(C(C)C)C1 c1(C(N2CC(OCCNC(CC(C)SC)=O)C2)=O)ccccc1-n1cccn1 N(C(=NCCC(C)C)NCC)C1CCC(C(=O)Nc2sccc2C)C1 C12CN(CC13CCC3)C2=O.CC(C)(C)CC(=O)N1CCCC1c1ncc[nH]1 C1(C2=CCOCC2)(CNC(=O)C(N2CCCC23COC3)=O)CC1 Cn1c(O)ncc(C(=O)NCCCCCN2CCN(C(=O)C(C)(F)F)CC2)c1=O c1(OC)ccc(C(N2CC(NCc3ccc(C)[nH]3)C3(CC3)C2)=O)cc1S(N)(=O)=O CN1CCC2(CCCN(C(=O)C(N)Cc3cc(Br)no3)C2)C1 N1(C(C=C(C)C(C)C)=O)CCC(C2(NC(=O)CC3(O)CCCC3)CC2)C1 n1(CC(=O)NC(C(C)NC(=O)CC2CN(C)C2)(C)C)cc(P(C)(C)=O)cn1 c1(NC2C(C)CSC2)nc2ccccc2nc1N1CCN2CCOCC2C1 C12(NC(c3occ(C)c3C)=O)CCOCC1CN(C(c1cc(Cl)ccc1N)=O)C2 c1(C(=O)NCCC(=C)CNC(=O)C(CC)CC(C)C)nc2c(Br)cccn2n1 N1(C(c2cc(C(F)F)no2)=O)CCN(C(=O)C(O)CN2CCCC2)C(C(F)(F)F)C1 C1(C(=O)Nc2nc(Cl)ccc2Br)CCCC12CCN(C(c1ccncc1Cl)=O)C2 Cc1nc(C(=O)Nc2ccc(C(=O)O)cc2Br)ccc1C(F)(F)F C1(NC(C=Cc2n(C)cnc2)=O)CC2CC1CN(C(c1cnccc1Cl)=O)C2 C1(N(C(=O)CCOC2CCC2)C)CCCN(C(=O)CC2CCSC2)C1 C1(C(=O)NC2CC(c3ccccc3)(NC(=O)C=CBr)C2)C(F)(F)C12CCC2 C1(CCNC(C2C(C)C2)=O)CN(C(C2CC3(CC3)C2)=O)CCS1(=O)=O C1(CNC(C2N(CC)CC2)=O)CN(C(c2cn(C(C)C)nn2)=O)C2CCCCC12 Cc1c(C(N2CC3C(CNC(=O)C(O)C(C)C)C3C2)=O)cccc1N C1(C(C)(C)NC(CC=CCC)=O)CCNC(=O)C1.C12=CCN(CC1)C2 N1(CCC)C(=O)NC(c2ccc3c(c2)C(=O)OCC3)C(C(=O)OC)=C1C1CCCC1 C1(NC(=O)CCSC2CCCC2)CCN(c2ccc(Cl)cc2)C1=O CC(CNC(=O)CCn1cccc1)C(F)C(=O)Nc1ccc(O)c(Cl)c1 C(=O)(CCC(F)(F)F)NC1C(CC)CN(C(=O)CCNC(=O)C=CCl)C1 N1(CC(C2CCC2)OC)CC(O)(CNC(c2cnon2)=O)C1 n1(CC=C)cccc1C(=O)NCC1CC1NC(C1CC(C)=NO1)=O Cc1ccc(COC(c2c(O)cc(Cl)cc2F)=O)cc1[N+](=O)[O-] C1(CCC(=O)NCC2N(C(CC)=O)CC2)CCCN1C C1(CNC(C2(SC)CN(C(CC)=O)C2)=O)CCN(C(=O)C2CC2)CC1 c1(C(N2CC3C(NC(C4CCC(C)(C)C4)=O)(C3)C2)=O)cnn2c1SCC2 C1(O)(CN(C)CCN2CCNC2=O)CCCN(C(=O)C(c2ccc(O)nc2)C)C1 C(=O)(CCP(C)(C)=O)NC(C)CN(C(=O)Cc1cncs1)C c1(CNC(C2(NC(C(CC=C)NC(=O)OC)=O)CCC2)=O)cc(C)cc(C)n1 c1(NC(C(CC)(C)O)=O)ccc(NC(=O)Cn2cccnc2=O)cc1C CCC(C)(C(=O)NC(C)(CNC(C1CC(C(=O)OC)C1)=O)C1CC1)C(F)F C1(C(=O)NCC(CNC(c2cnc(COC(C)(C)C)s2)=O)F)CCNC(=O)C1 Cc1ccc(CC(=O)NCc2ccccc2CN(C)C(c2nonc2N)=O)cn1 c1(-c2scc(C)n2)cccc(C(=O)NC(Cc2ccc(Br)cc2)C(=O)O)c1 N1(C(C=C)=O)CCOC2(CCN(C(c3cn(CC(=O)N(C)C)nn3)=O)C2)C1 C(=O)(C(C(C)C)c1cccc(OC)c1)NCCN(C(C1C(C=C)CC1)=O)CC C1(NC(C(C(C)O)C)=O)CC2(CCCN(C(C3(O)CC4CCC3C4)=O)C2)C1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC1CCCC(CNC(CCC#CC)=O)C1 c1(C(=O)NCC(CC)NC(c2cnc(C)n2C(F)F)=O)cncc(N)c1 c1(OCC)ccc(CC2CC(C(=O)N(C)C(C)C)C2)cc1Br N1(c2snc(COC)n2)CCC(C)C(NC(c2cnn(C(C)C)c2)=O)C1 c1(CC(C)OC)nc(-c2coc(SC)n2)n(-c2ccc(SC)cc2)n1 N1(C(C(CC=C)NC(C2Cc3nccn3C2)=O)=O)CCC(N(C)OC)CC1 c1(CNC(C2C(O)CCN2C(c2ccc(Br)cc2)=O)=O)ccc(Br)c(Cl)c1 C1(NC(Cc2ncc(C(=O)OC(C)(C)C)cn2)=O)CC2CC(=O)C1O2 C(=O)(C1CCCc2cc(C#N)ccc21)NCC1(C(C)(F)F)CCC1 C=CCCC(C)(C)NC(=O)C=C=CC.C(C(C)SC)NC(=O)COCCOC C1(C(=O)NC(C=C)C(C)C)CC12CCN(C(C1CCN(CC)CC1)=O)CC2 C1(NC(C(N2CCOCC2)C)=O)CC(C)(NC(=O)C(C2CC2)C2CC2)C1 c1(SCC)ccc(C)cc1F.N1(C(C2(N)CC2(C)C)=O)CCCC(c2c[nH]nn2)C1 N1(C(c2c(C)c[nH]c2)=O)C(C(=O)NC2C=CCCC2)CCC12CC2 N1(C(CC2N(C(C(OCC)O)=O)C3C2CCC3)=O)CC2CC1CS2=O.OC N1(C(=O)NC2CCCC2Cc2cnncc2O)CCOC(Cn2ccnc2)C1 C1(C)(NC(c2cnc(C(=O)OC)s2)=O)CCCC1NC(c1ccco1)=O N1(C(CCc2scc(C)c2)=O)CC(NC(=O)CC2CC3CCC2C3)C(F)(F)C1 c1(C(CNSn2cc(C3(N4CCCC4)CC3)nn2)SC)scc(C)c1C c1(NC2C3CN(C(c4c(C)ccc(NC(C)=O)c4)=O)CC32)ncc2c(n1)CCC2 Cc1ccc(C(N2C3CCC2(CNC(=O)CC(C)CN(C)C)CC3)=O)c(O)c1C c1(CNC(=O)NCc2ccc(-c3nn[nH]n3)cc2)cc2cccc(Cl)c2cn1 c1(C(N2CCN(C(c3cnsn3)=O)C(C(F)(F)F)C2)=O)ccc(Br)c(F)c1 N1(C(C(F)=CC)=O)CC(NC(=O)CNC(C)=O)CC(C)(C)C1 C1(CC(=O)NCCOC2CCN(C(=O)C3=CSCS3)CC2)CCS(=O)(=O)C1 C1(C(=O)NC2C(CNC(c3ncccc3F)=O)CCC2)Cc2nccnc2C1 c1(OCC)ccc(C)cc1C.C1(=O)CCC(=O)NC(C)C(=O)N(C)C(C)CCN1 N1(C(c2occ(C)c2)=O)CCC(C(=O)NCc2nc(C)sc2C)C12CCC2 c1(CNC(N2CCC(Cn3cncn3)C2)=O)cccc(CCF)c1 N1(C(COCCCN=[N+]=[N-])=O)CCCOC(C(=O)Nc2nc(OC)ccc2Cl)C1 c1(CNC(C=CC(CC)C)=O)ocnc1C(=O)N(CC(C)(C)O)C C1(NCCSC)CCN(C(=O)Cc2sccc2Cl)CC1F c1(C(N(C2CN(C(CCCc3ncc(C)o3)=O)C2)C)=O)cc(Cl)cc(Cl)n1 CC1(C)CC(CNC(C2OC3CCC2CC3)=O)CN(C(c2ccc(Cl)cn2)=O)C1 Cn1cc(-c2cc[nH]n2)c(C2CCC2C(=O)NCC(O)Cc2ccccc2)n1 O=C(C1CCCc2nn[nH]c21)NCC12CCC1CN(C(C1(F)CC1)=O)C2 c1(SC)nc(C)cc(=NCC(C2CC2)NC(=O)CCN2CCCS2(=O)=O)[nH]1 C(=O)(CC(C)N=c1[nH]c(=NC2C=CCCC2)[nH]c2c(F)cccc12)NC C#CCC(C)C(=O)N(CCCCCNC(=O)C(C)C)C N1(C(c2c(CC)cncc2)=O)CC2CCC(N(C(=O)Cn3ccc(C)n3)C)C2C1 C12(NC(C(CSC)OC)=O)CCC(CNC(C3OCCN(C)C3=O)=O)(CC1)OC2 C(=O)(C(CC(C)C)n1nnnc1-c1ccc(OCC(C)OC(C)=O)cc1C)OC C1(OC)CC(CNC(C2C(CC)CCC2)=O)N(C(=O)Cc2nonc2C)C1 N1(C(C(CC=C)NC(C)=O)=O)CCC2CCCC12C(=O)NCCC1CCCO1 c1(C(=O)NCCCn2cc(-c3c(OC)[nH]c(=N)cc3)nn2)c(F)ccc(C)c1Cl C(c1cnccc1C)=CC(N1CCC(N(C(C(COC)O)=O)C)CC1)=O c1(CCC(N2C(CNC(=O)C(O)c3ccsc3)CCC2)=O)cccc(Cl)c1 N1(C(C(C)n2ccnc2)=O)CC2(C1)CN(C(C1(C)CC(C3CC3)=NO1)=O)CCO2 N1(C(C2CCCN(CCC)C2)=O)CC2(CC2)CC1CNC(=O)C(C)CC(F)F Cc1cc(-c2cn(CCC(O)C(=O)N3CCC3CS(N)(=O)=O)nn2)nc(Cl)c1 C1(NC(CCOCC)=O)CCN(C(=O)COCc2ccncc2)CC1OC CC(C)(C)C(C(=O)N1CCC(NC(c2ccco2)=O)CC1)C(O)C(F)(F)F C1(NC(C(C2CC(F)(F)C2)OCC)=O)CCC(N(C(=O)C(O)CF)C)CC1 C1(CNC(=O)CCc2cnc(O)[nH]2)CN(C(=O)CC2(O)CCOC2)CCO1 N1(C(C=CSC)=O)CCOCC(CNC(c2cnnc(C)c2C)=O)C1 N1(C(Cc2ccc(C)cc2C)=O)CC2COCC2(C(=O)N(C)CC2CCOC2)C1 CCC(C)CCCC(=O)NCC1CC1NC(=O)COCC(c1ccccc1)C C(=O)(CC(C)CC(C)C)N1C(C(=O)NC(c2nc(C)sc2)C)CCC1C(C)C c1(OC)cccc2cccc(C(=O)NC3CN(C(=O)C4=CCCS4)CCC3O)c12 Nc1cc(C(N2CCCC(CCCCNC(C3CCCC3)=O)C2)=O)cc(O)c1Cl c1(C(=O)NCCCCN(C(C(C2CCCOC2)OCC)=O)C)ccc(O)c(N)n1 c1(C(=O)NCCCNC(Cc2ccc(OCCC)cc2)=O)cccc2nsnc12 C1(NC(C=Cc2cn(C)nc2)=O)CN(C(=O)CCCN=[N+]=[N-])C2(CCCC2)C1 N1(C(CC)=O)CCC2(CCCN(C(C3CCOC(C)C3)=O)C2)C1 C1(C2CCC2)(C(=O)OC)CCN(C(=O)C(=O)NC2CCC(N)CC2)C1 C1(C(=O)NC(CN(C(=O)Cc2cc(C(F)F)no2)C)(C)C)CCC(C#N)C1 c1(C(C2(C)CCCO2)NC(=O)COCCc2cccs2)ccc(C(F)(F)F)cc1 C1(C(=O)NC2(c3ccc(C)cc3)CC2)CCCN(Cc2ccc(C#N)nc2)CC1 Cc1ccc(C(=O)NC2CN(C(=O)CS(=O)(=O)N(C)C)CCC2F)cc1Cl CC1(C)CCc2cc(C(=O)NCC3CC3CNC(=O)Cc3ccccc3)ccc21 N1(C(CC=CCNC(C(COCC)N=[N+]=[N-])=O)=O)CC2(COC(=O)N2C)C1 C1(C(=O)NCCc2nc(C)oc2)NCCC12CC2(F)F C1(C2CCN(Cc3ccnc4ncnn34)CC2)(NC(C2CC=CCC2)=O)CC1 C1(N(C)C(C2CC(F)(F)C2)=O)CC2CCC(C1)N2C(=O)C(C)(C)Cc1cnn[nH]1 N1(C(c2cn3cc(C)sc3n2)=O)CCOC2CN(C(C3OCC3(C)C)=O)CC12 CN1CC(CO)CC1=O.c12cccc(n1)SCCNC(=O)CNC2=O CCCC(O)C(=O)NC1CC(NC(c2cccc(C)c2)=O)C(O)C1 N1(C(c2c(C)c(Cl)ccn2)C(=O)NCC2CCCO2)CC2CCCCC2C1C C1(NC(c2cn(CC)nc2)=O)CCN(C(=O)C2=CC(O)CCC2)CC(O)C1 N1(C(C(C=C)OC)=O)CC(CC(=O)NCc2ccc(C)nn2)C(C)C1 Cc1cc(C)c(C(=O)NCC2CC(NC(=O)CCS(N)(=O)=O)C23CCC3)c(O)n1 C1(CNC(C(=O)N(C)CCOCC(F)(F)F)=O)CCCCC1N1CCCC1=O CCCCC(=O)NCC1CCC1NC(C1COC(C(C)C)C1)=O CN1CC(C)(C(N2CCCC(C)(C(=O)NCc3cc(Cl)no3)C2)=O)CC1=O CCCC(C)CCCC(=O)N1CCC(CN(C)C(c2nc(Cl)c(Cl)s2)=O)C1 N1(C(c2c(C)ccc(C)n2)=O)CC2(C)CN(C(c3ccccc3)=O)CC2(C)C1 N1(CC(=O)N(CCOC)C(C2CCCCC2)=O)CC2CCC(O)C2C1 Cc1nn(C)c(C)c1CC(C)C(=O)NC(C)CN(C)C(C12CC(C)(C1)OC2C)=O C1(NC(=O)Cn2cc(Cl)cn2)COC2(CCN(C(c3cc(O)nc(O)n3)=O)C2)C1 Cc1sc(C(c2nnnn2CC(F)F)NCc2nc(C(C)(C)C)cs2)c(Br)c1C C(N=c1[nH]c(=NCC2CCC3(CC3)C2)[nH]c2ccsc12)C1(C)CCCCC1(F)F C1(C(=O)NC(CC=C)C)CN(C(=O)CCc2csnn2)CC(C)O1 C(c1cocn1)=CC(=O)NC1CC1CNC(=O)CC1COC(=O)C1 c1(NC(C23C(CN(C(c4cc(Cl)c(Br)c(Cl)c4)=O)C2)C3)=O)cccc2ccncc12 N1(C(=O)N(CC2(C)N=N2)C2CC2)CC2CCCC(=O)NC2C1 N1(C(N2CC3CC3(Nc3ccncn3)C2)=O)CC2CCCCC12 C12(C(N3C(C)(CC(=O)Nc4cn(C)nc4Cl)CC3)=O)CCCC1CCC2 C1(CC(=O)NCC(C)(C(C)C)NC(c2c[nH]nc2F)=O)(CC)CCOCC1 Cc1cccc(Br)c1C(C(N1CCN(C)C(C)C1)=O)NC(c1cccn1C)=O c1(C(=O)NCC2(O)CN(C(C(C)(C)C)=O)C2)cncc2c1CCNC2=O c1(C(N2C(C)(CC(N3C(COC)CC3)=O)CC2)=O)cc(C)cc(C)n1 c1(OC)cccc(-c2nc(-c3ccsn3)n(CCC(F)(F)F)n2)n1 C(C)(CC(C)C)(C(N)=O)NC(C1COCCN(C(CCSCC)=O)C1)=O N(C1CCCc2ccoc21)C(C(CCCNC(c1cc(CC)no1)=O)O)=O S(=O)(=O)(c1ccc(N2CC3CCC(C2)C3O)c(C#N)c1)N(CC(O)CF)C Cc1c(C(N2CCC(NC(=O)CCc3ccoc3)CC2C)=O)cc(N)cc1O C(=O)(C1CCCc2c[nH]nc21)Nc1ccc(CN2C(=O)NC23CCCC3)cc1 C1(NC(C2CC23CCSCC3)=O)CCCN(C(c2c(F)cccc2Cl)=O)CC1 N1(c2nc(C)nc(Cl)c2)CC(C)CN(C(C2CC(F)(F)C2)=O)CC1C C(=O)(CC(C)CC(C)(C)C)NCCCCCCC(=O)NC(C#C)C1CCC1 c1(CC)nnsc1C(=O)NC(C)(C)C(=O)NC1CC(CCC(=O)OC)C1 c1(SCCNC(=O)NCc2cnc(SC)s2)cc(F)ccc1F C(CC(C(C)C)NC(=O)CSc1nncs1)N(C(CCC=C(C)C)=O)C C1(NC(C(C)NS(CC)(=O)=O)=O)CC2C1CCN2C(=O)CC1CC(F)(F)C1 Cc1c(C(=O)NC2CN(C(=O)C(C)N(C)C)CCC2C(F)(F)F)cccc1O C(=O)(CCCCC(N)=O)NCC1N(C(C2C(C)(C)COCC2)=O)CC1 c1(CC(=O)N(C(C)CNC(c2ccc(C)cc2C)=O)CC)ccc(O)c(Cl)c1 c1(N2CC3C(CNC(C4(OCC)CCC4)=O)C3C2)[nH]cnc2nc(Cl)cc1-2 Cc1n[nH]c(C)c1CC(=O)NCC1(NC(C2COC(=O)N2)=O)CCC1 c1(SCC(=O)NC(CC(C)NC(C2(CC)COC2)=O)C)ccc(F)cc1 c1(C(=O)NCC(c2ccc(Cl)cc2Br)OC)cc2c(C(F)(F)F)cc(O)nc2o1 C(=O)(C1CCCc2nnn(C)c21)NC1CC(N(C(C=CCCC)=O)C)C1 CC1(C)OCCC1(O)C(=O)NCC1(C(N2CCC3(CCO3)C2)=O)CC1 N1(C(C(C)C)=O)CCC(C)(C)C1CC(N1CCSCC1C)=O C1(CNS(NC)(=O)=O)CCCN(C(c2cn(-c3cccc(Cl)c3F)nn2)=O)CC1 N1(C(CC2C(C)=NOC2=O)=O)CCC2CN(C(=O)C(C)(C)C3CC3)CC2C1 C(=O)(CC(C)(C)C(F)F)N1CC(CC(C)(C)C)N(C(=O)C(=O)NCC(F)F)CC1 C1(C(=O)NCC2(O)CCCOC2)(COC)C=CCN1C(c1sccc1OC)=O c1(C(=O)NCC2C(CC(=O)NCCCCC(=O)OCC)C2)nnc(O)nc1O CC1CCCCC1(CNC(=O)Cc1ccc(F)cn1)NC(=O)Cc1nc(=N)[nH][nH]1 c1(CC)ccc(C(=O)NC(c2ccc(C)cc2)CNC(C2CCCCO2)=O)cn1 N1(C(C=CCC2(NC(C3CC(=C)C3)=O)CCC2)=O)CCC(SC)CC1 C(=O)(C1(C)CCCc2ccccc21)NCCCCC(C)NC(C1C(C)=C1)=O C=CCC(C(=O)NC1CC=C(C(N2CCCC(F)(F)CC2)=O)C1)C(C)C S(=O)(=O)(c1c(F)cccc1F)NCC(C(=O)NCc1c(C)cccc1O)C C1(C(=O)NC(C2CCCCC2)CC)CC2CN(C(=O)Cn3cnc(C#N)n3)CC2C1 C1(CC(=O)NCC(CC)NC(=O)C(=O)CCC(C)C)CSc2ccccc2NC1=O C1(CNC(C2(CN(C)C)CC2)=O)CC(NC(c2ccc(O)cc2F)=O)C12CCC2 Cc1ccc(C(N2CCCN(C(=O)CCC3CC3C)CCC2)=O)c(N)c1C C1(NC(C(COC)O)=O)CN(C(c2ccc(Cl)cc2Br)=O)CC12CCC2 N1(C(COC(C)=O)=O)CCOC2(CCN(C(c3cc(Br)c(C)c(Br)c3)=O)CC2)C1 Cc1csc(C=CC(N2CCN(C3CCN(C(=O)Cn4ncnn4)C3)CC2)=O)n1 c1(OC)ccc(F)c(C(=O)NCCC2(NC(C3CCOCC3(C)C)=O)CCC2)n1 c1(C2C(C)(C)C2)nc(-c2cnccc2I)n(C2CCCSC2)n1 C1(COC)(CNCc2cncc(C(=O)N)c2)CCOCC1 C(=O)(C(C)CC(N)=O)NCCN1CCN(C(C(C(C)OC)N(C)C)=O)CC1 C1(C)(COC)CCN(C(=NCC2CCC2)NCC2(CC(N)=O)CCCCC2)C1 Cc1ccc(C)c(COc2cc(Br)ccc2OCC(=O)Nc2ccccc2C)c1 C1(NC(c2c(CC)ocn2)=O)CCCCC1C(=O)NCC(C)C(F)F CC1(C)CCN(C(C2(C#N)CCCCC2)=O)C1C(=O)NC1CCCC1O C1(C)(C(N2CC3C(CNC(CCNC(=O)OC)=O)(C3)C2)=O)CC(C2CC2)=NO1 N1(C(C2C(=C)C2)=O)CCC(CCNC(=O)CC2(CSC)CC2)C(F)(F)C1 c1(C(=O)NCC2(C)N(C(c3ccc(SC)o3)=O)CCC2)cncc2cnccc12 C1(OC)CN(C(c2cc(-c3ccco3)on2)=O)CC1NC(C12CC3CC1C2C3)=O C1(C(=O)NC2CN(C(Cc3cn(C(C)C)nc3)=O)C(CO)C2)CC12CCOCC2 Cc1cnc(C(C)NCC2(CC(=O)O)CC2)s1 C1(CNC(CN(C)C)=O)CN(C)CCN1C(c1sccc1Cl)=O C1(c2n(CC)nnn2)(NCCc2nc(C)no2)CCC2CN(C)CC12 c1(-n2cc(C3CCCN(C(c4cccnc4CO)=O)C3)nn2)c(F)cccc1Cl N(C1CCc2cc(CNC(c3cc(C4CC4)ns3)=O)ccc21)C(C(C=C)(C)O)=O c1(C(=O)NCC(=C)CCNC(C2CC2(C)C)=O)ccc(Cn2cccn2)cc1 N1(C(C(C)N(C(C)=O)C)=O)CCn2c(CNC(=O)C3=C(C)CCCC3)nnc2C1 c1(C(=O)NCCCC(C)NC(=O)Cn2nnnc2C2CC2)ccnc(Cl)c1Cl n1(CC2N(C(=O)NC3(CS(C)(=O)=O)CC3)CCC2)cc(Br)cn1 N1(C(c2ccc(CCC=C)cc2)=O)CC2(COC(CNC(=O)COCCF)C2)C1 CC1CC(=O)N(c2ccc(Br)c(C(N)=O)c2)C1=O C1(NC(c2cc(COC)[nH]n2)=O)COC2(CCN(C(c3cccc(CO)n3)=O)C2)C1 C1(NC(=O)CCC2CCC3(CCC3)C2)CCC12CN(C(=O)NCCON1CCCC1)C2 c1(C(=O)N(CC2CCN(C(C)=O)C2)C2CC2)ccc(OC(F)(F)Cl)cc1 C(=O)(C(C)CC(F)(F)F)NC1C(CNC(C2(F)CC(C(=O)OCC)C2)=O)C1 c1(CN(C)Cn2cc(-c3ccc(C4CC4)cc3)nn2)cccc(F)n1 C1(S(N)(=O)=O)(c2cn(CCC3CC(NC(C(c4ccc(C)s4)C)=O)C3)nn2)CC1 C1(NC(c2ccc(OC(C)(C)C)cc2)=O)CCC12CN(C(c1ccnnc1)=O)C2 C(C(C)(C)C(=O)NC1CC2(C1)CC2NC(c1[nH]nnc1C1CC1)=O)NC(C)=O C1(N(C(=O)COCCc2cccs2)C)CCC(NC(C2CC3C=CC2C3)=O)CC1 c1(CNCC=CC(=O)Nc2cncc(F)c2)cccc2ccccc12 N1(CC(=O)C2CC2)CCC(CO)C1.C1(C(=O)C(CCOCC)C2CC2)CC(=C2CC2)C1 c1(N(C(Cn2cc(CNC(C3(OC)CCCCC3)=O)nn2)=O)C)cccn(C)c1=O Cc1ccc(NC(=O)NC(c2ccc(F)c(C3CC3)c2)CN(C)C)cc1Cl c1(NC(CC2CCN(Cc3cc(OC)cc(F)c3)CC2)=O)ccc2nccn2c1 c1(C(N2CC(NCC3(C(=O)OC)CC(=C)C3)C2)=O)c(C)cc(F)cc1C c1(NC(c2ccc(N3CCCCC3)c(Br)c2)=O)ccc(Cl)cc1[N+](=O)[O-] c1(C(N2CCC(C)(NC(C3(C)N(C)CCC3)=O)CC2)=O)cnn2c1NCCC2 C1(CC(=O)NC2COCCC2NC(C2(CO)CCC2)=O)CCCCC12CC2 C1(NC(CCC=C)(c2nnnn2C2(C)CC2)C2CCCO2)CS(=O)(=O)C12CCCC2 c1(OC)ccccc1C(C)(C)C(=O)NCC(C)N(C(=O)COc1ccon1)CC Cc1cc(C(=O)NC(C)C(=O)N2CCC2C(C)(C)O)oc1C c1(C(=O)NC2CC(CNC(C3CCC(=C)CC3)=O)C2)ccc(F)c(Cl)n1 Cc1nn(CC(=O)NC2CC(C(F)F)(NC(c3ccc[n+]([O-])c3)=O)C2)c(C)c1C C#CCC(C)(CNC(=O)C(C)(C1CC1)N(C)C(C1CCC(=O)N(C)C1)=O)CO CC(CCC(=O)NCc1cncc(CO)c1)NC(=O)C(C)c1ccsc1 n1(CC(N2CCC(C)(c3cn(C4CCCC4)nn3)C2)=O)cc([N+](=O)[O-])cn1 C(=O)(C(CN(C)C)NC(C1CC1C(F)(F)F)=O)NCC#CCOC c1(CCCCC(=O)NCCC2CCN(C(=O)C=CBr)C2)ccc(F)c(F)c1 C#Cc1ccc(C(N2CC(CO)OC(CC)C2)=O)c(F)c1Cl c1(OC)ncc(Cl)c(C)c1C(=O)NCC1CN(C(=O)C(C)C2CC2)CCC1(F)F C=C1CCC(C(=O)NC2C=CCN(C(c3cc(C(C)CC)no3)=O)C2)CC1 C(=O)(C(C)(C)C(=O)NCc1ccc(C(=O)NCc2ccco2)nc1)NC c1(C(C)C(=O)N(C2CCN(C(C3CCC(=O)N3)=O)CC2)C)ccc(F)c(F)c1 C12(CC(=O)NCC(C)CNC(=O)CSCc3ccc(Cl)s3)COC(CF)(C1)C2 c1(C(=O)NC2C(C(N3CC(C(=O)OC)OCC3)=O)C2)ccc2nccn2n1 C(CCCCC(=O)N1CC(N2CCN(C(=O)CSc3cnn(C)c3)CC2)C1)OC N1(C(C(C)(C)OC)=O)CC2CCC(C1)N(C(c1cc(Br)oc1C)=O)C2 c1(CCC(N2CCC(C(C)NC(C3CC(C(N)=O)C3)=O)C2)=O)ccc(O)nn1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N(C(C)CN(C)C(c1c[nH]nc1C(F)F)=O)C c1(C(=O)NCCN(C(C(CO)N(C)C)=O)C2CC2)ccc2ncnn2c1 C1(C(N(CC(=O)NC2(CO)CCCCC2)CC2CCC2)=O)C=CC=CC=C1 c1(C(=O)NC(C2(O)CN(C(=O)Cn3cccn3)C2)C)cc2cc[nH]c(=O)c2s1 CC1(C)CC(=O)NCC1C(N1CC(OCCNC(=O)CC2CCCC2(F)F)C1)=O C(=O)(C(CC)CC(C)C)NCC(N(C(C(C)OCC=C)=O)C)C1CC1 C1(C(N2C(C=CC(NOC(C(=O)OC)C)=O)CCC2)=O)CC2(COCCO2)C1 c1(C(C(=O)NC(CNC(c2ccn(CC(C)C)n2)=O)CO)C)nc(F)ccc1Cl CCC(F)(F)C(C)(C)NC(C1CN(C(C2CC(=O)NC2(C)C)=O)CC1(F)F)=O Cc1cc(Cl)cc(C(N2CC(CCNC(C3(C4CC4)CC3)=O)C2)=O)c1C C(N=c1ccnc(NCc2c[nH]nc2C(C)C)[nH]1)c1c(C)c2c(s1)cccc2 Cc1c(C=CC(N2CC(NC(=O)C(C)(F)F)C(C)(C)C2)=O)cnn1C c1(NC(=O)NC(c2cccnc2)CO)ccnn1C1CCCCC1 N1(C(c2occ(C)c2)=O)CCN(C(c2ccc(Cl)o2)=O)CC1c1cn[nH]c1 C1CC(O)C(=O)N1.C1(C(=O)NCC2CC(NC(C)=O)C2)C(C)C1(F)F.C(C)(=O)CN C(=O)(C(CC(C)C)C(C)C)NCC(CN(C(C=C(CCN(C)C)Cl)=O)C)C Cc1cccc(C(=O)NCC2(NC(=O)CCc3ccsc3)CCOC2)c1C c1(C(N2C(C)CCC(NC(c3cncn(C)c3=O)=O)C2)=O)cc(O)cc(C#N)c1 N1(C(c2c(C#N)nc[nH]2)=O)CCCN(C(=O)CCN2CCCC2)CCC1 Cc1nc(C)n(CCC(=O)NC(C)(CNC(=O)Cc2ccsc2Cl)C2CCC2)n1 C1(C(=O)NC2CCC(NC(c3cnc(C(C)=O)s3)=O)CC2)(COC)CCC(=O)N1 N1(C(COCC(=C)C)=O)CCC2CCN(C(=O)C(C(C)C)n3cnnn3)CC12 C(=O)(C#CC1CCCC1)NC12CCC(NC(C3C(C)(C)CCCO3)=O)(CC1)C2 C(CNC(=O)C1=CCSC1)(CC(F)(F)F)NC(=O)C(O)C(F)F C1(CCC(N2CCC(NC(C3CC(CN(C)C)C3)=O)C2)=O)CCCCCC1 CC1(CN(C(C2CC2c2ccccc2)=O)CCl)CCCN(C(=O)C2=COCCC2)C1 CCCC(C#N)C(=O)NC(C)(C)CCNC(C1CCC(C(F)(F)F)CC1)=O c1(CC(C)C)ncc(C(N2CCCC(CN(C)C(C34CC(O)C3C4)=O)C2)=O)n1C N1(C(COc2ccc(C(C)=O)cc2)=O)CCCC(C2CCCC2)C1 N1(C(c2ncc(F)cn2)=O)CC2CCC1C(O)C2O CN1CCN(CCC(=O)NCC2CC2NC(=O)C(C2CCCCCC2)O)CC1 Cc1ccc(CN)c(OCC(F)(F)F)c1.C(C)(C)(CN(C)C)SC C1(C(N2C3C(C(=O)OC)C(C3)C2)=O)CN(C(C2CC2(C)C(F)F)=O)CC1(F)F c1(CN(CC(=O)NC2CCN(C(CC3(C(=O)OC)CC3)=O)C2)C)ccccc1Cl N1(C(C(C(C)C)C)=O)CC2(CCCC(CNC(C3CN4CCC3CC4)=O)O2)C1 C1(C(N2CCCC(NC(C(C)CCO)=O)(CO)C2)=O)CCCC(F)(F)CC1 C1(C(N2CCC(C(C(=O)NC3(CC(C)C)CC3)F)C2)=O)CN(C)CCO1 C(=O)(C(C)(O)C(C)(C)C)NC(C(C)NC(=O)COC(C)(C)C(F)(F)F)(C)C C1(CC)CN(C(=O)CSCC2CC2)CCC1NC(=O)C(CC1CC1)CC1CC1 C(CNC(=O)COC1(C)CCC1)(CC(=O)NCC(CO)C1CC1)OC C(CCCCC(=O)NC1(C(=O)N(CCC(C)O)C)CC1)=CC Cc1nn(C)c2sc(C(=O)NCC3CN(C(=O)CC45CC(C4)C5)CCC3C)cc12 C12(NC(=O)CCCF)CCCC1CN(C(c1cccc3nn[nH]c13)=O)C2 c1(C(=O)NC2CC(C)(NC(=O)CSc3cccs3)C2)cccc(C(N)=O)n1 C1(NC(COCCC=C)=O)CCCN(C(c2cc(N)ccc2O)=O)CC1 N1(CC)CCC(C(=O)NC2CN(C(C3(C(=O)N(C)C(C)C)CC3)=O)C(C)C2)CC1 C(=O)(CCCS(C)(=O)=O)NCC(C)(CC(C)C)NC(c1cc(C(C)=O)c(C)nc1)=O Cc1ccc(C(=O)NC2(C(N3CCCOCC3)=O)CC(F)C2)nc1O c1(OC)cccc(CCC(=O)NC(C)(C)CN(C)C(c2ccnc(OC)c2)=O)n1 c1(C(N2CC3CC(NC(c4n(CC)cc(Cl)c4)=O)C3C2)=O)c(C)nc(O)nc1C C1(C)(CNC(C2CCCN(C)C2)=O)CCC(NC(=O)CC2CCCCCC2)CC1 C1(C(=O)NC2CC(C(=O)NCCn3c(C)ccn3)C2)CNC(=O)CC1C c1(CC(N2CC(NC(CSCC=C)=O)C3C2C3)=O)ccc2nc[nH]c2c1 c1(OC)cc(C(=O)NCC2C(C)CCN2C(c2n[nH]c(C)c2O)=O)nn1C CCCC(C)(C)CC(=O)N1CCC(CCOC)(NC(C2CCOC2C2CC2)=O)C1 c1(C(N2CC3C(NC(c4cccc(C)c4N)=O)C3C2)=O)cc(F)c(F)c(F)c1F c1(C(=O)NCC2C(C(N(C)CC3(C)CCCO3)=O)C2)cccc(=O)o1 Cc1nc(C)c(C(=O)NC2(CCCNC(c3ccc(C(C)C)o3)=O)CC2)o1 c1(SC)nc(N2CCC(N(C)C(c3ccc(Cl)nc3Cl)=O)C2)cc(Cl)n1 c1(C(=O)NC2CCC(CNC(C3(F)CCCC=C3F)=O)CC2)cc([N+](=O)[O-])cs1 C(=O)(C(C)=NOCC#N)NCC(C(N1CCC(OC)CC1)=O)OC C1(C(=O)NCC2CCN2C(C2(CC(F)(F)F)CC2)=O)NC(=O)C2CC12 N1(C(C(C)N(C(C)=O)C)=O)C(CC(=O)NC(C2(O)CCCCC2)C)C2CCCC12 CC(C)CCCCCNC(C1CCCCN(C(c2ccoc2)=O)C1)=O CCCC(C)(CC)C(=O)NC1CCCC1C(=O)NC(C)CCC(C)(C)C Cc1cccc(-c2ccc(C(=O)N(C3CCCC3)Cc3cccnc3)s2)n1 N1(C(COCC)=O)CCOC2(CCN(C(C3CC3C)=O)C2)C1 C1(NC(=O)Cn2nnc(=O)[nH]2)CN(C(c2ncsc2Br)=O)CC12CC2 C(C)(C)(CCCNC(=O)CSCc1cccc(Cl)c1)NC(C1C(C)(C(C)C)C1)=O C(=O)(C(C)=Cn1ccnn1)NCC(CC)(C)NC(=O)CNC(c1cnoc1C)=O c1(-c2n(C(CC)C)nc(Cc3cnn(C)c3)n2)cccn1C(=O)OC CC(=O)CCC(=O)N1CC(OCCC(=O)NCCC2(CO)CCC2)C1 C(CCC(C)C)OCC.N12CC(C1)NC2=O.C1(C2CCCC2)CCN1 C(=O)(C(C)CC(C)(C)C)NC(C(=O)NCCc1scc(C)n1)CC(F)F Cc1c(Cl)ccnc1C(N1CCC(N(C)C(c2cc3[nH]ccc3s2)=O)C(C)C1)=O C1(NC(C=C(C)Cl)=O)CCOC12CCN(C(C1CC3CCCC(C1)C3=O)=O)CC2 C1(CNC(C2(F)CCCC2)=O)CC2(CCN(C(C3(Cl)CC34CCC4)=O)CC2)C1 Cc1cc(=NC2CCC(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2)[nH]c(Cl)n1 C123CC(CN1C2=O)C3.c1(CNC(C2C(=C)C2)=O)cnn(-c2ccccc2)c1CC C=CC1(O)CN(C(C2CCCC2NC(=O)C(O)CSC)=O)C1 CC(C)(C(=O)N1CC2CCC(C1)N2C(=O)CCCC(=O)c1cccs1)C(F)(F)F c1(CC(N2CCC(N(C(=O)C=CC3CC3)C)C2)=O)cccc(Br)c1 CN(C)S(C)(=O)=NS(=O)(=O)NCc1cc([N+](=O)[O-])ccc1Br c1(CC)ccc(CNC(CC(C)C)c2cccs2)o1 CC(C)C(O)C(=O)NC(C)CCC(=O)N1CC(NC(N)=O)C1 C1(C(C(=O)N2CC(C(=O)N(C)C)C2)NC(C(=O)NCC)=O)CCCCC1 C12CCN(C1)C2=O.C1(COCCC)C(CO)C1(C)C.C(=O)(C(O)C1CC1)N N1(C(C(CC)N(C)C)=O)CCCC(NC(c2occc2F)=O)C1 Cn1nc(Br)c2ncnc(-c3nnc(SCC4(C)CCS(=O)(=O)C4)o3)c12 Cc1cn2cccc(C(=O)NC3CN(C(=O)CCOC4CCCC4)CC3C)c2n1 c1(C(N2CCC(CCNC(COCC(=O)OC)=O)C2)=O)cc2nnn(C)c2s1 C1(CC(=O)N(CCCN(CC(=O)N(C)C)C)C)CC2CC1CC21CC1 c1(C(=O)NCC(CC=C)NC(c2cnc(C)s2)=O)nc(O)[nH]c(=O)n1 c1(CC(=O)NC2CC(N(C(C3CC(OC(C)=O)C3)=O)CC)C2)nccn1C Cc1cnsc1C(=O)N(C1(CC(N2CC(O)(c3cnn[nH]3)C2)=O)CC1)C CC1CCNCCC1N1CCCCNC1=O.c1(C)cccc(O)c1.c1(N)cn[nH]c1 C#Cc1cncc(C(=O)N(CC(O)CN(C)C(c2c[nH]c(Br)c2)=O)C)c1 C(=O)(CC(CNC(=O)CCOC1CCC1)C1CCC1)N(C1CCCCC1C)CC C1(NC(c2cc(C)nc(C)c2)=O)CCSC12CN(C(C1CCC(=O)N1C)=O)C2 C(=O)(CCC(=O)c1cccc(F)c1)NCC1CN(C(Cn2c(C)ccn2)=O)C1 c1(C(N2C(CC)C(NC(c3cnn(C(F)F)c3)=O)CC2)=O)ccc(Cl)cc1F C(C(=O)NCC(CO)NC(c1cc(N)cc(O)n1)=O)(c1ccccc1)=C(C)C c1(C(N2CC(NC(CC3(CSC)CC3)=O)C(O)CC2)=O)cc(N)c(F)c(F)c1Cl C1(C(N2CC(OCC#C)C2)=O)CC12CCN(C(C13CCCC1C3(F)F)=O)CC2 C1(NC(C(COCC)NC(c2cn(C)nc2SC)=O)=O)CC2C(CO)C2C1 CC1C2C(CCN2C(C2CCCC2C2CC2)=O)CN1C(=O)Cc1ccc(Cl)cc1 C1(CC)C(NC(=O)CC2CC3CC3C2)CCCN1C(c1cc(OC)nc(OC)c1)=O c1(CNC(C(C)(C)NC(=O)NCC)=O)cccc(O)c1F.C1CCCC(=O)N1 C12(C(=O)NC(C(=O)NC(C=C)CO)(C)CO)C(=O)C3CC1C2C3 C1(CNC(c2ccccc2)=O)CN(C(c2cnc(Br)s2)=O)C2CC12 CCC(CC)C(=O)NCC(=O)NCC(=O)NC1CC(CF)C1 c1(C(=O)NC2CCN(C(C3N(CC)CC3)=O)CC2C)cnn2c1CCCN2 c1(C(=O)OC)oc(C)nc1C=CC(N1CCC(OCc2ccncc2)C1)=O c1(OC)cnc(Cl)nc1N1CCCC1(C)CNC(=O)COCc1cccnc1 O=C(CC(C(F)F)c1ccccc1)NCC12CC(NC(C3CC3C(F)F)=O)(C1)C2 C(C(C)(C)CC(=O)NC(C)(C)CN(C)C)NC(C1(CCCC)CCCC1)=O c1(C(N(C)CC2CN(C(C(C)OCC=C)=O)C2)=O)coc(C2CCCC2)n1 c12nc(cs1)CN(C(=O)CCCc1ncco1)C2.n1(CCC(=O)O)cc(Cl)cn1 C1(NC(c2ccc(-c3cccnc3)cc2)=O)C2COCC1CN(C(C1CC1F)=O)C2 NC1CCC=C1C(=O)N1CCCC1Cn1cc(CN2CCCCC2)nn1 CC1C(C(N2CCC(F)(CNC(C3(c4cc[nH]n4)CCC3)=O)C2)=O)CCN1C N1(C(COC(CC)C)=O)CC(NC(=O)CSc2ccc(Cl)cc2)CC12CCC2 c1(C2(CNC(c3cn(CC)nc3)c3nnnn3C)CC2)ncccc1F N1(C(c2c[nH]nc2F)=O)CCCC(N(C(=O)CCc2ccc(=N)[nH]c2)CCO)C1 C1(CC)CN(C(=O)COCC(=O)NC)CC1CC(=O)N(C)OCc1ccccc1 CCCC(C(O)C(=O)NC(CC)C(=O)N(C)C)NC(=O)COC C(CC1c2ccccc2CCN1C(=O)OC)C(=O)OC(C)(C)C.C1(C)C(=O)N1 N1(C(c2coc3c2CN(C(C(C(CC)O)C)=O)C3)=O)CCC2(COC(C)C2)C1 N1(C(C2C(C(=O)OCCC(=O)NC3CC4CCC4C3)C2)=O)CCCN(CC)CCC1 N1(c2ncc(C#C)cn2)CCC2(CCCCC2NC(c2nc(CCC)no2)=O)C1 c1(C(N2CCN(CC(C)NC(c3cncn3C)=O)CC2)=O)cccnc1Cl C(=O)(C1=CC2CCCC12)NCC1CCCN(C(c2c(CC)occ2)=O)CC1 C(CC(C)C)(C(=O)N(CC(C)C(=O)NC)C)N(C(C1(CC)CC1)=O)C c1(CC)ccc(C(=O)NC(C)(CNC(c2cc(CSC)[nH]n2)=O)C(C)C)c(C)c1 C(N=c1[nH]c2c(c(=NC3CC3C)[nH]1)SCC2)c1c(C)ccc(C)c1 c1(OCC)ccc(C2CCCN2C(=O)C(C)(C)n2ccc(C)n2)nn1 N1(CC=C)CCC(N2CCSCC2CCNC(=O)CC2C=CCCC2)C1=O C1(CC(N2CC(O)(C(C)NC(=O)CC3OCCCO3)C2)=O)COCC(C)(C)O1 C1(NC(c2nc(CC)oc2C)=O)C2CCN(C(c3cc(C(C)C)n(C)n3)=O)CC12 N1(C(CNC(c2ccoc2)=O)=O)CC(O)C(O)C1CNC(C1CCC=CCC1)=O CC1(C)CCN(C(=O)C(F)=C2CCC2)CC1NC(C1CCCC1C(F)(F)F)=O CC(C)(C)C1=NOC(C)(C(=O)NCCC(O)C(F)F)C1 c1(CC)cccc(C)c1-n1nc(-c2cnn(C)c2)nc1C(n1ccc(Br)n1)C CC(C)CC(C)CC(=O)NC1CCN(C(c2nocc2Br)=O)C1C1CC1 c1(CC)c(C(=O)NC(CNC(=O)CCCn2cncn2)C(C)C)nnn1C Cc1nc2ccc(C(N3CCN(C)CC3CNC(=O)C(F)(F)CC3CC3)=O)cc2s1 c1(NC2CC3CN(C(c4nn(CC)c(C)c4)=O)CC3C2)ncnc2c1ccn2C c1(NC(C2N(C(CCCC(C)C)=O)C(C)CC2)=O)ccc2c(c1)CC(=O)N2 C(=O)(C(O)C(C)(C)C)NCCC(C(=O)OC)NC(C1(COC)C2CCC12)=O CCC(O)(CC(=O)NCC1CCC1CNC(=O)CCP(C)(C)=O)c1ccccc1 C1(CNC(C2(C#N)CC2)=O)CCCC(NC(c2cccc(O)n2)=O)C1 C1(C(=O)NCC2CCN(C(c3n(C)c(S)nn3)=O)C2)CN2CCC1CC2 C1(NC(C(CCCC)C)=O)CCC2CC1CN2C(C12COC(CCO1)C2)=O Cc1cccc(CC(=O)N(C2CCN(C(=O)C(c3ccccn3)O)C2)C2CC2)c1 CCC(=O)CCC(=O)NC1CC2(C1)CC2C(=O)N(CCCO)C CC1(C)CCN(C(=O)C2=COCCO2)CC1NC(c1ncc(Cl)cc1F)=O Cc1nn(CCO)c(C)c1C(=O)NCCCC1CCCCN1C(=O)C(O)C1CC1 c1(C(=O)NCC(C)CN(C)C(c2ccnnc2S)=O)cc(C#N)on1 C=CCC(CC)C(=O)N1CC(C(=O)NCCNC(C2CCCC(F)C2)=O)C1 CC(C(O)C(F)F)NC(C1(NC(=O)CC2CCCNC2=O)CC(O)C1)=O c1(CNC(CN(C(C2C(C)C2C)=O)CC)=O)ccc(O)cc1 Cc1ccc2c(=O)c(C(N3CCC(C4CCCN4)C3)=O)cn(C)c2n1 C1(C(=O)NC(CNC(c2cn(CCC)nc2)=O)C2CC2)CCc2nnnn2C1 N1(C(C=C(COC)C)=O)CC(CNC(c2c(C)noc2C)=O)OC2(CCC2)C1 c1(OC)ccc(CN2CCN(C(=O)C(C)=O)C3CC23)c2ccccc12 N1(C(CC2CN(C)C2)=O)CCC(C2CCCN(C(=O)C=CBr)CC2)CC1 C1(NC(c2ncn(C)n2)=O)CCSC12CN(C(c1ccc([N+](=O)[O-])cc1)=O)C2 N1(C(CC(c2ccccc2Br)N(C=O)C)=O)CC(=O)NC(=O)C1.C(=O)C1=CCSC1 c1(N2CCC(NC(C(C)n3ccnc3)=O)C(C)(C)C2)ncc2c(ncn2C)n1 C1(NC(C2CC(CC(F)F)C2)=O)CC2CCC(C1)N2Cc1nc(Cl)ccc1Cl C(C)(CCC(=O)NS(C)(=O)=O)NC1CN(C(=O)CCOC2COC2)C1 N1(CC)C(=O)CCC1CC(=O)N(C1CCN(C(=O)C=CSCc2ccco2)C1)C C=CCCCCCC(=O)N(CCCN(C(=O)CN1CCC(F)(F)C1)C)C c1(C(N2CCC(C(C(N3CC(CC#C)OCC3)=O)C)CC2)=O)cncn(C)c1=O O(NC(=O)CC(C)CNC(c1cc(C#N)ccc1C)=O)C(CC)CC c1(C(N2C(CC(=O)N(CCCCC=C)C)CCC2)=O)cc(C(F)(F)F)nn1C Cc1oc(-c2ccccc2F)nc1CC(=O)NC(C)CNC(c1cnn(C)c1)=O c1(CC)ccc(C=CC(=O)NC2CCC2NC(C2(C)CCCCC23CC3)=O)cc1 c1(C(N2CCCCC(N(C(C3OCC(C)C3)=O)C)C2)=O)cnc2ccccn12 N1(C(C=CCN(C)C(C2CC(F)(CF)C2)=O)=O)C2CCCC1COC2 C1(C(=O)NCC(C)(C)NC(c2ccc(SC3CC3)cc2)=O)CC12CCSCC2 C1(CC(=O)NC(C(=O)N(CC#CC)CC#C)Cc2ccoc2)CCCOCC1 C(=O)(C(C(C)O)NC(C1CCCC1CNC(c1cc(=O)cc[nH]1)=O)=O)OC c1(SC)nc(N2CCCC(NC(C34CCOC(C)(C3)C4)=O)CC2)c(C)c(Cl)n1 CC1=C(C(=O)NCC(O)CN(C(=O)C(C)Oc2cccc(C#N)c2)C)CCO1 C(CCCC1CC1)(C(=O)NCC1CCOC1)N(C(=O)CN1CCOCC1)C Cc1nccnc1C(=O)NCC(C(C)(C)C)NC(c1cc(Br)no1)=O C(C(CC(=O)N=c1cc2n([nH]1)CCCC2)OC)NC(C(C(=C)C)(C)C)=O C=C(C)CC(C(=O)NCCOCCCO)NC(c1ccns1)=O C1(C2CCN(C(=O)C(C)O)C2)(NC(Cn2c(C)ccn2)=O)CC1 c1(C(=O)NCC(C2CCOC2)NC(c2c(C(C)C)nns2)=O)nccc(Cl)c1F c1(C(=O)NCC=C(C(=O)NC(C=C)C2CCC2)C)ccc(CO)s1 CC(CCC(=O)N1CCC(NC(c2ncn(C)n2)=O)C1C(C)(C)C)N(C)C c1(C(=O)NC2CCN(C(=O)C(F)OC(F)(F)F)CC2F)c(F)ccc(F)c1Br C1(NC(CC=CCCCCC)=O)CCOC(C(N2CCC2CC(C)C)=O)C1 CCCC(C)(CC)C(=O)NC1CC(C)CN(C(C2CCN(C(=O)NC)CC2)=O)C1 C(CCC(=O)NC1CCC1NC(C1(C)CCOC1)=O)OCC C1(C(=O)NC(C)CCC(C)C)(CC)CCN(C(C2CCC(C)C2)=O)CC1 C1(NC(=O)OCC)CCCC1NC(=O)C(Cc1cccnc1)N(C)C C1(NC(C2C(C)OCC2)=O)(CF)CCN(C(=O)CC2COCCOC2)C1 c1(C(=O)NCC(C2CCOCC2)NC(=O)CC2CC2)c(F)cccc1Cl C1(CC=CC(=O)NCC(C2CC2)NC(=O)Cn2ccnn2)CCOC1C1CC1 C1(CC(=O)N(CCC(C)NC(=O)CCc2ccc[nH]2)C)(COC)CCC1 c1(C(=O)Nc2ccc(NC(CS(CC)=O)=O)c(C)c2)ccc(C#N)c(C)n1 CC(C)CC(CNC(=O)CC1OCCCO1)NC(=O)COc1ccccc1F c1(CC)nn(C)c(CC(N2CC3C(CNC(=O)C(O)C4CC4)C3C2)=O)c1Cl c1(C(N2C(CCNC(C(CSC)OC)=O)CCC2)=O)cc(O)c(F)cc1N n1(CC)ccnc1CN(C(=O)CN(C(c1ccc(Cl)s1)=O)C1CC1)C c1(OC)nccc(C(=O)NC(C2(O)CCN(C(=O)CNc3cccs3)C2)C)c1F C1(CC(=O)N(C2CCCN(C(=O)CCC3OCCO3)C2)C)NC(=O)CNC1=O c1(CNC(C(=O)NC(C)Cn2ccnc2)=O)ccc(Cl)nc1 c1(C(N2CCC(CN(C(C3(CSC)CC3)=O)C)CC2)=O)cc2c(nn1)CCCC2 C=CCCCCC(=O)NC1CC(OC)CN(C(C2(C)CCCO2)=O)C1 Cc1c(NC(N2CCOC(C(F)(F)F)C2)=O)cnn1-c1ccccc1F Cc1ccc(C(N2CCCC2C(C)NC(=O)CCF)=O)nc1C C12(CC)CCC(NC(=O)CSCCC(=O)OC(C)(C)C)(CO1)C2 c1(C(N2CC(CC(N3CC(C)(CO)C(O)CC3)=O)C2)=O)c(F)cc(C#N)cc1F c1(CC(=O)NC(CNC(C2CC2F)=O)C2CCC2)c(Cl)cccc1Br N1(C(C(CC)SC)=O)CCn2ncc(CNC(C3(S(N)(=O)=O)CCC3)=O)c2C1 C1(NC(C2CN(C(=O)C3CC3)C2)=O)C=CCN(C(=O)CCOC2CCCOC2)C1 CC(C)(C(=O)N1CCN(C2CN(C(C3CCCC3C3CC3)=O)C2)CC1)C(F)(F)F C1(NC(CC(=O)OC)=O)CC2CCC1N2C(c1cn(Cc2cccnc2)nn1)=O c1(C(=O)NCC2N(C(CCC3CCC(C)O3)=O)CCC2)c(Cl)oc2ccccc12 CN1CCCC(NC(C2CSCN2C(C2OC3CCC2C3)=O)=O)CC1 C(C(CO)(CO)NC(c1ccsn1)=O)N(C(C(c1ccc(F)cc1)CC)=O)C C1(Sc2scc(C(N(CCCC)CCO)=O)n2)CCCN(C(=O)OC(C)(C)C)C1 c1(N2CCC(O)(C(C)NC(c3c(C)cc(F)s3)=O)C2)cc2nncn2c(C)n1 C1(NC(c2c(CC)nns2)=O)CCCC12CCN(C(=O)CN1CCCC1C)CC2 C1(=O)CCC(=O)NC2CN1C2.N1(C(C(C)Nc2scc(CC)n2)=O)CCCC(C)C1 c1(CC(N2CC(C=C)C(NC(c3nc(C)oc3C)=O)C2)=O)c(O)nc(=N)[nH]c1C c1(C(C(=O)NC2CC(F)(F)C2)N(CC)Cc2ccc(F)cc2)ccc(C#N)o1 C(=O)(CC(C(C)OC)NC(=O)Cc1ccoc1C)NC(C=C)C c1(CN2C(C(=O)Nc3ccc(F)cc3Br)CSCC2)cc(F)c(Br)cc1F c1(C(N2CCCC(C)(CNC(c3n(C)ncc3)=O)C2)=O)ccc2c(c1)OCCC2 Cn1nc2ccccc2c1C(=O)NCC1CC(NC(=O)CN2CC=CC2)CC1O CC1COCC(CC(=O)NCC2CCC2C(N2CC3CC2(CN(C)C)C3)=O)O1 Cc1nsc(CNC(=O)C=CC(C)NC(=O)C(C)N2CCCC2)n1 c1(C(NOCC(=O)NC(C2CCCCO2)C)=O)sccc1CO C1(COC)CN(C(=O)C(O)CSC(F)(F)F)CCN1C(C1CC(=C2CC2)C1)=O c1(C(=O)O)cnnc(CCC2CC3CC2CN3)c1.n1(CCC=O)ccccc1=O CC1CN(C(C23CCC(CC2)OC3)=O)CCN1C(N1CC(C(N)=O)CCC1C)=O N1(C(C(C)Cn2ccnc2)=O)CC(F)(F)CC1C(=O)NCC(C)(C)C CC1CCN(C(C2CC(F)(F)CN2C(=O)Cc2cccnc2)=O)CCS1 C(=O)(C(C)CC(C)C(C)=O)NC(CC)CC(=O)N1CCC(C(F)F)C1 Cn1sc(C(=O)NC2CCCN(C(=O)CCCc3ncco3)C2)cc1=O n1(CC)cccc(NC(C2(OC)CCN(C(=O)C(O)CC(N)=O)C2)=O)c1=O N1(C(CCSCC(N)=O)=O)CC2CC1CN2C(c1cnc(CC2CC2)nc1O)=O C(C(C(C)(C)C)NC(=O)Cc1cncc(F)c1)NC(c1c(CC)csc1)=O N1(Cc2n(CC)nnn2)CC=C(CCNC(=O)Cc2ccc3ocnc3c2)CC1 c1(C(=O)NC2CC(F)(CNC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)cc2n(n1)CCC2 N1(C(CCCCC#C)=O)CC2CN(CC(=O)NC(N)=O)CC2C1 CC1(C)C(=O)CC1C(=O)NC1CCC(CNC(c2ccncn2)=O)CC1 C1(OC)CCC(CC(=O)N(CCCNC(=O)C(C)(F)F)C2CC2)CC1 CN1N=C(C(=O)NCCN(C)C(c2ccnc(-n3ccnc3)c2)=O)CCC1=O Cc1cc(N)cnc1C(=O)N(C(CC(C)C)C(=O)NC1C(C)CCCC1C)C CC1(C)COCC(C(=O)NCC2=CCN(C(=O)CC3CCCO3)CC2)C1 C(=O)(CCCCC(C)(C)C)N1CCC(N2CCN(C(CC(=C=C)C)=O)CC2)CC1 C1(C(=O)NC2(CO)CC2)(COC)CCCN1C(c1coc(C(N)=O)n1)=O C1(C(=O)OC)CCN(C(C2(CN)CCC2)=O)C2CCCCC12 c1(C(N(C(c2cccc(OC)c2)CC)C)=O)ccc(N)c(-n2ccnn2)c1 c1(N2CCC(COC)(CNC(c3cccs3)=O)CC2)cc(C#N)ccc1[N+](=O)[O-] N#Cc1cc(C(=O)NC23CC2CN(C(c2ccc(C(N)=O)cc2)=O)C3)on1 c1(OC)ccc(OCC(=O)OC(C)CO)c2ccccc12 N1(C(C(CCC)(C)CC)=O)CCC2(C1)CN(C(c1csc(CC)n1)=O)CCO2 C(C1=CCCN(C(=O)CC2CC3(CC3)C2)C1)NC(=O)Cc1cnc(C2CC2)[nH]1 C1(C(N(C(CC(=O)OC)C)C)=O)CN(C(C2CC(=O)N(C)C2)=O)CC1C(C)C N1(C(CCSCCOC)=O)CC(C(=O)NCCCCF)CCC1C C1(C(=O)NC(C#C)CC2CC2)CCC(C)CN1C(c1coc(C2CC2)n1)=O CCC(C)(C)CC(=O)NCC(C1CC1)NC(=O)C(C)C(C)c1ccccc1Cl c1(NCC(=O)NCC2(O)CN(C(COC3(C)CCCC3)=O)C2)cc(O)ccc1O C1(CNC(CC2(C#N)CC2)=O)CC2CCCC2N1C(c1coc(Cl)c1)=O C(CCCC(=O)N1CC2CC1C2)N(C(C1(C(=O)OCC)CCC1)=O)CC n1(CC(=O)NCC2CC(NC(C(C)n3cnnn3)=O)C2)nnc(-c2ccco2)n1 C1(c2nc(C(F)(F)F)on2)(Nc2cc3ccccc3cn2)Cc2ccccc2C1 C(CN=c1[nH]c2c(c(=NCc3nc4c(s3)COCC4)[nH]1)CSC2)=CCOC c1(C(N(C)CC2(O)CCN(C(C3C(=C)CC3)=O)C2)=O)cc(=N)[nH]c(Cl)n1 C12(C(=O)NCCCN(C(=O)COC3CCCCC3)C(C)C)CCCC(C1)OC2 c1(CNC(CC)CC2CC2)nc(C2CCOCC2)no1 C#CC1CC(NC(c2ccn(CCNC(=O)CC3CCC(=O)C3)c2)=O)C1 c1(OC)ccc(C(N2CC(NC(=O)CN3CCC(C)(O)C3)C(C)C2)=O)cn1 N#CC1CN(C(c2ccc3nonc3c2)=O)CCN1C(c1ccc(CO)nc1)=O Cc1cc(Cl)cc(C(=O)NC(C)C(C)NC(=O)C=Cc2ccncc2)c1N C=Cn1nccc1C(=O)NCC1CCC(NC(c2cccc(COC)n2)=O)C1 c1(N2CCC(NC(=O)C=CBr)C(F)C2)ncc2c(n1)CCOC2 C1(N(C(C(COC)O)=O)C)CCC2CN(C(=O)C(C)Oc3cccc(C)c3)CC12 Cc1cc(CCC(=O)NCC2CCC2NC(c2oc(C3CC3)nc2C)=O)c(C)s1 C(=O)(C(CN=[N+]=[N-])NC(C1OCC2CCCC12)=O)N(C)CC1CCC1 CC(C(=O)N1CCCC1C(C)NC(=O)CN1CCCC1)C(F)(F)C(F)F N1(CC(=O)C(c2csnc2Cl)=O)CC2CC2C1.C(CCN(C(=O)C1CC1)C)N CC(=O)CCCC(=O)N1CCCC(CN(C)C(c2ccc(C)c(O)c2)=O)C1 CC1COC2(C1)CN(C(=O)COC(C)(C)CNC(=O)CCC1CCCO1)C2.C(C)(=O)O c1(NC(C)=O)no[nH]c1=NC(=O)C1CCN(Cc2sc(Cl)nc2Cl)C1 c1(C(N(C)CC2CCN(C(C3CCC(C)O3)=O)CC2)=O)cnc2ccccc2c1 Cc1nc(O)nc(C)c1C(=O)NC(CNC(C1CC(C(C)(C)C)C1)=O)CC(C)C CCCC(CC)C(=O)NC1CC1CNC(=O)CC(C)SC CC1CC(NC(c2ccncn2)=O)CCN1C(c1cnc(F)c(F)c1)=O C1(C(N(C2(CC(C)(C)C)CC2)C)=O)CCN(C(C2CC2C(C)(F)F)=O)C1(C)C C12(NC(C3C(=C)CC3)=O)CC(C1)N(C(C1CCCCN1C)=O)C2 CCCC(C(=O)NCC1CC(C)N(C(=O)Cc2ccc(C3CC3)cc2)C1)N(C)C Cc1cc(S(=O)(=O)N2CCCN(C(=O)C(c3cccn3C)=O)CC2)c(F)cc1Cl N12CCC(C(C)C1)NCc1cc(co1)C2=O.c1(OC(C)C)ccc(C(=O)O)nc1 C1(CN(C)C(C2C3CC4C(C3)C24)=O)C2CN(C(=O)CC3CC3C(F)(F)F)CC12 N1(c2ccc(OC)cc2)CCCC(NCc2nc(Br)c[nH]2)C1=O Cc1ccc(CCC(N2CCC(CNC(C3CCC3)=O)C(C)C2)=O)cc1Cl c1(CCC(C(=O)NC2CCCC2)N(CCF)CC)nc2ccc(F)cc2s1 c1(C(=O)OC(CCC#N)Cc2ccc(F)cc2)ccc([N+](=O)[O-])cc1 C1(NC(c2cc(C)no2)=O)CCN(C(c2ccc(OCCF)cn2)=O)C1(C)C C1(C(=O)NC(CNC(c2ccc(C3CC3)s2)=O)C2CC2)CCC2(CC1)CC2(F)F c1(C(N2C3CN(C(CSc4n(C)nnn4)=O)C(C3)C2)=O)scc2c1CCCC2 N1(C(CC(C)(C)c2ccccc2)=O)CC(NC(=O)C2=COCCC2)CC(F)C1 C=CC(C)CC(=O)NC(CC1CC1)C(=O)N(C)Cc1cccs1 N1(C(c2cc(C(=O)OC)oc2)=O)CCC(NC(C2(N(C)C)CC2)=O)CC1C1CC1 N1(C(C(CC#C)(C)C)=O)CCC(C2CC2NC(=O)COc2cnc(Cl)cn2)CC1 C#CCCCCCC(=O)N1CCCC(NC(=O)CCc2cc(C)on2)C1CC c1(C(=O)NCC(CC)NC(=O)CC2CCCC(C)C2)cc(C)nn1CC N#Cc1ncc(NCC2CC(NC(=O)CC3CCCC(F)(F)C3)C2)nc1C#N C(=O)(C1=C(F)CN(C(C2CC2Cl)=O)CC1)N(CC(C)C#N)C C(=O)(C#CC1(C)CCCO1)N1CC(N(C(=O)C=Cc2cocn2)C)C(O)C1 C#Cc1cc(C(=O)NC2C=CC(CC(=O)NCCC(C)(C)OCC)C2)ccc1C c1(C(=O)NC2CCOCC2NC(C2CCC2)=O)ccc2nc[nH]c2n1 c1(CNC(C(c2ccc(Cl)cc2)OC)C)ccc2c(c1F)OCCO2 c1(C(N2CCN(CCCNC(CC3(C=C)CC3)=O)CC2)=O)cccc(C)c1CC c1(OC)ccc2occ(C(N3CCCC3C(C)NC(=O)CC34CC(C3)C4)=O)c2c1 C=CCCCCC(=O)NCC1CCN(C(C2C3COCC23)=O)C1 C(CCC(=O)NC1CC(NC(=O)NCCn2cc(-c3ccn(C)n3)nn2)C1)=CC C1(CCNC(Cn2c(C)nc(C)n2)=O)CN(C(=O)C=CC2CCC2)CC(C)O1 C1(CNC(CCCCC=C)=O)C2CCCC1N(C(=O)C(C)S(N)(=O)=O)C2 c1(C(N(C2CN(C(C=C(C)Cl)=O)C2)C)=O)ccc2c(c1)CCCCS2 C(=O)(CN=c1[nH]c(=NCc2cc(Cl)ccc2OC)[nH]c2c(F)cccc12)NCC C=CCC(C)(CC)C(=O)N(CC(O)CNC(=O)CCCOCCC)C N1(C(CCCOC)=O)CCC(N(CCO)C(c2ccc(C)cc2)=O)CC1 C(=O)(C(O)C1=CCCCC1)N1CCC2C(C(=O)Nc3c(C)c(CO)ccc3)C2C1 N1(C(C(CC=CC)C)=O)CCCCC(NC(c2[nH]ccc2-c2ccccc2)=O)C1 C(=O)(C(F)CCC(C)C)NCC1(OCC)CN(C(=O)Cc2nccn2C)C1 C(C(C)(C)C(=O)NC1CN(C(=O)C(C)CSc2ccccc2)CC1O)SC N1(C(C(C)N(CCC)C(c2nnsc2N)=O)=O)CC2CCCC(O)C2C1 c1(OC)ccc(-c2nc(C(=O)NC3CC3CNC(c3n[nH]cc3C)=O)cs2)cc1 C(C)(C)(CCC(=O)NC(C)CS(C)=O)NC(C1ON=C(C)C1)=O C(N=c1cc(Br)[nH][nH]1)C1CCCN(CC(O)Cc2ccccc2)C1 Cc1ccnc2c(C(N3CC(CNC(=O)CCn4cncn4)C3)=O)cnn12 c1(CNC(CC2(N(C)C)COC2)=O)cccc(NCC2CCCN2C)c1 C1(C(=O)NCCCN(C(=O)C(C)CC2CC2)C(C)C)CN(C)C(=O)N1 c1(C(N(CCN(C(C(C)N(CC)CC)=O)CC)CC)=O)cnc(C)[nH]1 C(=O)(CCCC(N)=O)NCC(CC)NC(=O)Cc1cn[nH]c1 Cc1cn2ccc(C(=O)NCC3CN(C(=O)CSC(F)(F)F)C4CC34)cc2n1 c1(CC)ccc(NC(C2CCN(C(C3CCCC(SC)C3)=O)C2)=O)c(C)c1 N1(C(C23CCC(OC)C2C3)=O)CCC(NC(=O)C=C2CCC(C)CC2)C(F)C1 CC1=CCC(C(=O)NC2CN(C(c3ccnc(NS(C)(=O)=O)c3)=O)CC2C)CC1 C1(CNC(C2C=CCS2)=O)CC2(CC2)CN1C(c1cccs1)=O C1(C)(C(N2CC(CCC)OCC2)=O)CC12CCN(C(=O)CCC(=O)NC)CC2 N1(C(COCCCC)=O)CC(C2CCCN(C(=O)CNS(=O)(=O)N(C)C)C2)C1 C=CCC(CC)C(=O)NC(CCC)CC(=O)NC(COC)COC C(=O)(C(O)C(F)(F)F)N1CCC(N(C(c2cn(CC(F)(F)F)cn2)=O)CC)CC1 N1(C(=O)NCCC2CCCN(C)C2)CCCSCC1NC(C)(C)C CC1CN(C(=O)C=Cc2ncc[nH]2)CCCN1C(=O)C1=C(Cl)CCCC1 c1(OC)ccc(Cl)c(C(N2CCN(C(=O)CNC=O)C(CS(C)(=O)=O)C2)=O)n1 C1(c2ccccc2)(NC(=O)OCC)CCCN(C(=O)C(C2CC(F)(F)C2)OC)C1 CCC(C)(C)C(C)CC(=O)NCC1COC(C)(C)CN1C(=O)C1=CC2C=CC1C2 Cc1scc(C(=O)NCC2CCCCC2C(=O)NCCN=[N+]=[N-])c1C N(C1CCc2cccnc21)C(C1C(NC(c2cc(C)ncc2)=O)C1)=O C(=O)(C(F)CC(CC)CC)NC1C(C(NOCC=C)=O)C2CCC1C2 C1(CCNC(C(CC)C)=O)CCCN(C(C2CCCN2CC(C)C)=O)C1 CC1(C2CC2)CN(C(=O)CCCOCc2ccccc2)CCO1 C1(C(=O)NC2(CF)CCN(C(=O)CCc3ccc(F)cc3)C2)CC2CCC1CC2 C1(C)(COC)CC(NC(C2(CF)CC2)=O)CN1C(c1nc(O)c(C)s1)=O c1(C(=O)NCc2c(OC)nsc2)cncc(CNC(c2cccc[n+]2[O-])=O)c1 CCCC(C(=O)NCC(O)CCNC(c1sccc1C(C)C)=O)NC(N)=O c1(OC)ccc(CNC(=O)C(N2CC(C)OC(C)C2)=O)cc1OCc1ccccc1 C=CCCCC(=O)NC1CC1NC(=O)Cc1ccc(O)cn1 c1(C(CCO)NC(c2nnnn2-c2ccccc2)(COCC)C)cccnc1 c1(C(N2CC(N(C3CCN(C(c4cccs4)C)CC3)C)C2)=O)cc(C)nc(C)n1 C1(NC(c2ccc(SC)cc2)=O)CCN(C(c2cc(CO)ccc2F)=O)CC1F c1(C(=O)NC(C(=O)NC(C23CCC(CO2)C3)C)CCC2CC2)cccc(F)c1N N1(C(C(=Cc2ccccc2)NC(C)=O)=O)CC(NC(=O)CSC(C)C)CC(C)C1 C(CC(F)F)(C(=O)NCCN1CCC1)NC(c1c(OC)nsc1)=O c1(-c2nc(CCSC)nn2-c2ccn3nccc3c2)ccc(C2=CCCC2)cc1 CS(=O)(=O)c1ccc(N2CCCC(CNC(c3cc4ccccc4s3)=O)C2)nc1 C=CC1OCCC1C(=O)NCc1cnn(C)c1C(=O)NCC(C)(O)C(F)F C1(N(C(=O)C=CC(F)(F)F)C)CN(C(c2ccnn2C)=O)CCC1O C(=O)(CC(C)C(C)(C)NC(=O)OC(C)(C)C)NCCC(C=C)C CCC(C)(C(=O)NC1CCN(C(=O)CCc2cccs2)CC1O)C(N)=O CC1CCN(C(=O)CCc2cncc(F)c2)C1CNC(c1cccnc1)=O CN(C(=NCCCF)NCc1cnnn1C)C(=O)CC1COCCN1C N1(C(C(=O)NCCCCS(N)(=O)=O)=O)CC2(CCCC2)c2ccccc21 C1(F)(C(=O)NC(C)C(CO)NC(=O)Cc2cccc(F)c2)CCCOC1 C1(CNC(C2(C(C)C)CC2)=O)COCCN(C(=O)CN2CCC(=O)NC2=O)C1 c1(C(N(CCNC(c2cc(C)[nH]n2)=O)C2CC2)=O)ccc(F)c2cccnc12 C1(OCC)CCN(N2CCC(CN3CCOCC3)CC2C(N)=O)C1 N1(C(=O)CC2C=CCC2)CCC2(CCCN(C(=O)C3=CSCS3)C2)CC1 CCCC(C(=O)N1CCC(F)(C(=O)Nc2ccc(OC)c(C)c2)CC1)NC(C)=O N1(C(CCN(C(C)C)C(C23CCC(CC2F)C3)=O)=O)CCC2(CCOC2)CC1 C(CC(C(=O)NCC(C1CCN(C(C2CCNC2=O)=O)CC1)O)OC)SCC C(CCC(O)C(=O)NCCN1CCOCC1C)NC(CCOCCOCC)=O Cc1ccc(F)c(N)c1C(=O)NCCN(C(=O)C1=C(Cl)CC1)C1CCCC1 c1(C(N(CCCNC(C(CC#C)C)=O)C2CC2)=O)ccc(Br)c(C)c1N N1(C(C2CCC(=O)S2)=O)CCCCC1CNC(=O)C#CC1CC1 Cc1nc(C)c(C(N2CCN(CC(=O)NC3CCOC(C(C)C)C3)CC2)C)[nH]1 c1(OC)cc(CN2CCSC(C(N3CCCCC3C(N)=O)=O)C2)ccc1Br C1(C(N2CC(C)(NC(=O)CCc3ccc(Cl)s3)C2)=O)CC(F)C(=O)N1 Cc1nc(N2CCC(NC(c3n[nH]c(C)c3O)=O)C23CCC3)cc(C#N)n1 C1(CNC(C(N2C(CC)CCC2)=O)=O)C2CN(C(=O)CCC3CC3(F)F)CC12 C1(CC(=O)NCc2cc(C)no2)CCOC1(C)C.C12(CCC1)CC(=O)N2C C1(C(=O)NCC(CC)NC(c2coc(C(C)(C)C)n2)=O)CCC12CCC2 Cc1cc(N(C(c2ccccc2)=O)CC23CCC(CC2)N3)cc(N)c1Cl N1(C(C)C)CCN(N(CC(=O)Nc2cc(COC(C)(C)C)on2)C)CC1 c1(CCC(N2CCC(C(C)NC(=O)CC3CC3)C2)=O)ccc2ccn(C)c2c1 N1(C(C(CCC)N(C)C)=O)CCN(C(=O)Cn2nc(C)c(C)c2C)C(CCC)C1 C(=O)(C(CNC(c1cncn1C1CC1)=O)CC1CC1)NCC1(CC)CCOC1 c1(C(N2CCC(CCOC)(NC(C3(O)CC3)=O)C2)=O)n[nH]c2c1CCOC2 N1(C(C2C(CC)C2)=O)CCCCC2(CCN(C(c3cnc(OC)c(C)c3)=O)C2)C1 C1(O)(C(=O)NCCC2(C(N(C)CC3CCCOC3)=O)CC2)CCOC1(C)C N1(C(C2(C(C)C)CCN(C(CSCCCC)=O)C2)=O)CCCC(C)(CC)CC1 Cc1cc(NCC2CCC(NC(=O)C(O)CC3CC3)CC2)ccc1[N+](=O)[O-] N1(C(Cc2c(C)occ2)=O)CCC2(CC1)CC(NC(C1CCC(N=[N+]=[N-])C1)=O)C2 C1(O)(NC(CN(C)CC)=O)CCC(C)CC1.C12(CC1)CCN(CCOCC)C2=O C12(C(=O)NCC3C(NC(c4scc(C)c4C)=O)C3)CCCC1C2(F)F C1(C(NOCC(=O)NCCn2c(C)nnc2)=O)CCN(C)CC1 C1(C(=O)NCC(=O)NCC(=O)NC)(CSC2CCOC2C(C)C)CC(C)(C)C1 CC1CN(C(=O)CCOCCNC(C2COCC2(C)C)=O)CC(C2CC2)O1 N1(C(CC2CC(C)C2)=O)CC2CC1(C(=O)NCC1(N(C)C)CCCC1)C2 C1(N(C)C(=O)OC(C)(C)C)CN(C(=O)CC2CC(C(=O)O)C2(C)C)CCC1O Cc1c(NC(=O)NC2CC2c2ccn(C(F)F)n2)cccc1Cl N1(C(CC(C)C2CCCO2)=O)CC2(C1)CN(C(c1ccnc(Cl)c1Cl)=O)CCO2 O=C1CN(C(c2cnc(O)c(F)c2)=O)C(C(=O)NC2(CO)CC2)CN1 c1(C(C(=O)NC(CC)C)N(CC(C)(C)N2CCCC2)C)nc(Cl)cc(Cl)c1C c1(CNC(CC(C)N2CCCC2)=O)cccc(N2CCCC2)c1 C1(NC(C(C2CCCC2)OC)=O)CC(N=c2[nH]c3cc(Br)cnc3s2)C1(C)C C=CCC(C(=O)NC1C2CC(NC(c3cc(O)nn3C)=O)CC12)OC c1(OC)ccc(CC(=O)NC2CCC(N(C)C(c3cn(C)nc3Cl)=O)C2)c(F)c1 S(=O)(=O)(CCCS(=O)(=O)N(C)C)N(c1ncc(C2CCCCC2)cn1)C N1(C(c2c(C)ncc(N)c2)=O)CCC(C)N(C(C2CCC2(F)F)=O)CC1 c1(C(C(=O)NC)N(c2ccc(F)cc2)C(C)C)nc(Cl)sc1Cl.C1(N)CC1 CCCC(C(=O)N1CCCC1CN(C(=O)CCc1nc(C)c(C)[nH]1)C1CC1)OC Cc1ccc(O)cc1C(=O)NC(CO)CCC1CC1.c12cncc(c1)C(=O)N2 c1(OC)ccc(CNC2CC2C(=O)Nc2cncc(C(F)F)c2)c(O)c1 C12(C(=O)NC(CC=C)CNC(c3ccn(C)c3)=O)CCC(C)(CO1)C2 c1(OC)ccc(-c2oc(C)cc2C(=O)NC(C)CN(C)C(c2cncs2)=O)cc1 C1(C(=O)N(CC(O)CN(C(=O)CCc2cnoc2)C)C)(CC)CC(C)(C)C1 C(C(C)N=c1[nH]cnc2cc[nH]c12)N1CCN(OCCOC)CC1 c1(CNC(C(N2CCCNCC2)(C)C)=O)ccc(F)cc1.c1(CC(=O)O)ccc(F)cc1 c1(CC)sc(C(=O)NCCCOCCN(C(=O)C(O)CC2CCCC2)C)cc1C c1(CN(C)C(c2ccn(CC(F)F)c(=O)c2)=O)c2c(nn1C)CCC2 CC1CCCc2c(C(=O)NC3CCCCN(C(=O)C4=NOCC4)C3)cnn21 C1(CCN(C)C(C2CC2F)=O)CCCCN1C(c1cccc(OCC(F)F)c1)=O C1(C(=O)NC2(C3CCCN3C(c3ccc(C4CC4)nc3)=O)CC2)C2CCCCC12 c1(C(C(=O)NCC(Cn2cc(CCN(C)S(N)(=O)=O)nn2)OC)C)ccc(C)s1 C1(NC(=O)CCc2ccccc2)CN(C(c2cc(F)ccc2O)=O)C2CCCC12 N1(C(=O)Cc2csc(Br)c2)CCN(C(c2nn[nH]c2Cl)=O)C2CC12 N1(C(c2cc(C)nc(O)c2)=O)CCC2CN(C(=O)C(C)Cc3cnn(C)c3)CC12 Cc1oc2cc(C(=O)N(CC(C)NC(=O)C(N3CCCC3)C3CC3)C)[nH]c2c1C C(N=c1cc(C)nc(NC(c2nc(O)n[nH]2)C)[nH]1)c1c2cnn(CC)c2ncn1 C1(OC)CC(CCNC(=O)CC2(CSC)CC2)N(C(=O)CC(C)C)C1 Cc1cc(O)nnc1C(=O)N(C1CCC(NC(c2ccncc2C)=O)C1)C C1(N(CCCC(=O)Nc2ocnc2C)C(C)=O)CCCN(Cc2ccccc2)C1 N1(C(C23CC(CN(C(COCCC(C)C)=O)C2)C3)=O)CCC2CN(C)CC12 c1(NC(CN(C(=O)C=CCN(C)C)CC#C)=O)cnn2c1OCCC2 CC(C(C)(C)C(=O)NC1CC1(C)C(F)F)NC(c1c[nH]c(=S)cn1)=O N1(C(COC(CC)(C)C)=O)CCC(C(=O)NC2CCCC2COC)C(O)C1 c1(CNC(C2(CS(C)(=O)=O)COC2)=O)cnn2c1CN(C(C1CC1Cl)=O)CC2 n1(CC)nnnc1C(c1cncs1)NC(C)Cn1ccnc1C C=CC(C)(O)CC(=O)NCC1CCC(CNC(c2ccsc2CSC)=O)CC1 C(=O)(C1Cc2ccc(Cl)cc21)NCCN(c1nc(C)nc(=N)[nH]1)CCC c1(C(N2CC(NC(c3onc(C)n3)=O)C(C)C2)=O)cc2ncccc2s1 Cc1cccc(Br)c1C(=O)NCC1CCCN1Cc1ncc[nH]1 C1(F)(CN(C)C)CCN(C(C2(NC(C(C3CC3)OCC)=O)CCCCC2)=O)CC1 Cn1nnc2c1CCN(C(C1CN(C(c3ccn(CCF)n3)=O)CC13CC3)=O)C2 N1(C(CC(C)CF)=O)CCCC2CN(C(C3(CO)CC3)=O)CC12 CCCC(C(=O)OC)n1c(C2C3CN2C3=O)nnc1C.c1(SCC)ccccc1Br N1(C(CCC#C)=O)CC(O)CC1CNC(c1ccc(OCC)cc1)=O CCS(=O)c1ccccc1C(=O)NCC1CC1NC(c1cccc(C(C)C)c1)=O c1(C(N2CCC(CN(C(C)=O)CC)CC2)=O)ccc(S(=O)(=O)NC)o1 c1(OC)nc(C)ccc1C(=O)NCCC1(CNC(=O)CCC2CCOC2)CC1 c1(N2CC(SC)C(O)C2)ccc(N2CCCC2)cc1[N+](=O)[O-] c1(CC(CNC(=O)Nc2ccccc2Br)CO)ccc(OC(F)(F)F)cc1 C=CC1(C(=O)NCC(C)(C)CCNC(c2ccc(C(N)=O)o2)=O)CCOCC1 C=C=CCCC(=O)NC1CC1CNC(c1ccc(CO)s1)=O.C(CC)CC N1(C(CC)C)CCN(C(=O)COCCNC(C2CNC(=O)O2)=O)CC1 C12(C(=O)NC3CN(C(C=Cc4c(C)ccnc4)=O)C3)CCC(C)(CC1)OC2(C)C N1(C(c2ccc(CC)[nH]2)=O)CC(C2CN(C(C3CC4CCCC4C3)=O)C2)C1 C1(NC(C(F)=CCC)=O)CCN(C(c2ccc(OC)cc2F)=O)CC(C)(C)C1 c1(C(=O)NC(C)(C)C)ncc(C(=O)NCC=CCNC(C2C(C)CCC2)=O)cc1Cl N1(C(C(c2ccc(C)cc2)O)=O)CCCCCC1C(C)(C)C(=O)O CCC(CC(=O)NCC1(F)CN(C(=O)C=Cc2ccccc2C#N)C1)C(C)(C)C c1(C(N2C(C(=O)NC(CC=C)C)CCC2)=O)ccc(C)nn1 Cn1cnc(C(=O)NCCC(Cc2ccccc2)NC(=O)CSC2CC2)n1 c1(C(N2C(C)CCC(NC(CC(=O)NC)=O)C2)=O)nn(C)c2c1CCC2 c1(C(C(C)C)OC)nc(CO)nn1-c1cncc(Br)c1 CCCCC(O)CC(=O)N1CCOC(C(C)NC(=O)CO)C1 c1(C(=O)NCC(CNC(N)=O)O)cnc(CNC(C2CCNC2=O)=O)nc1 CC1CN(C(=O)C(C2CCOCC2)F)CCN1C(=O)C(F)OC(F)(F)F C1(C(=O)NCC2CCCC(NC(=O)CC3(O)CCCC3)C2)CC2(C1)CC(F)(F)C2 N1(C(c2csc(C)c2C2CC2)=O)CC2CCC(NC(C3CCCC3)=O)(C2)C1 c1(C(=O)NC(C)C(=O)NCCN2CCC3CC23)c(Cl)cnn1C N1(CC)CCOCC1CC(N1CCCC1CNC(c1cc(Br)c[nH]1)=O)=O C#CC1CCC(NC(C2(C(N)=O)CCC2)=O)C1.c1(CO)cccc(C)n1 c1(C(N2CCC(CNC(C3(CC4CCC4)CC3)=O)CC2)=O)cc(F)ccc1F Cc1c(C(N2CCCCC(CNC(=O)CCC(C)(C)N(C)C)C2)=O)cccc1O N1(C(CCCn2cc(COC(C(C)O)=O)nn2)=O)CCCCC1Cn1cccn1 C(=O)(C1=NOC2(CCOC2)C1)NCC(CNC(c1c(F)ccc(C)n1)=O)(C)OC Cc1cc(C(=O)NC2CCN(C(=O)CCc3cc(C)on3)C23CC3)cc(C)n1 N1(C(=O)NCC(c2ccc(C)cc2C)(C)C)CCn2c(CC(C)C)nnc2C1 CC(C)C(C(=O)NCC1CN(C(=O)C(C)CO)C2(CCC2)C1)C(C)C Cc1ccnn1CC(N1CCC(CN(C(=O)COCc2scnc2C)C2CC2)C1)=O C1(C(=O)NC(CCCNC(c2c(C)cnn2C)=O)C)CCN(CCO)C(=O)C1 C1(CNC(C(COC)C)=O)(NC(=O)CCc2ccnn2C)CCCCC1 N1(C(C2N(C(=O)C(O)C3CC3)CCC(=C)C2)=O)CCCC2(CCC2)C1C CCC(C)CCCCC(=O)NCC1(C(=O)NCC(=O)N(CC)OC)CC1 CC1CCN(C(C(Cc2ccc(Br)cc2)CC(F)F)=O)CCS1=O n1(CC)ncc2c(N(C)CCC3CCN(C(c4oc(C)cc4C)=O)C3)ncnc12 Cc1cc(C(N2CC3(NC(=O)C(C)SC(F)(F)F)CCC2CC3)=O)c(O)c(C)c1 c1(CNC(c2ncccn2)=O)nc2c(s1)CCN(C(C1C=CCC1)=O)C2 C12(C(N3C4(CNC(c5ccc(F)c(Cl)n5)=O)CC(C3)C4)=O)CCCC1C2(F)F c1(CNC(C2CC(CN)C2)=O)cc2cc(Br)ccc2s1 c1(C2C(C(=O)OC)C2C(=O)OC)ccccc1NC(=O)OC(C)(C)C C1(CNC(=O)CCOC2CC2)CN(C(c2nc[nH]n2)=O)CCCO1 C(=O)(C1c2ccccc2C2CC1C2)NCC1CCCN(C(C(C(C)C)SC)=O)C1 CCCC(C)CC(=O)N1CCC(C(=O)NCCC)CC1C C1(c2c(C(=O)NCC3CCC(F)CC3)c[nH]n2)CCCCN1CC=CC(F)(F)F Nc1ccc(-c2cn(CCCCCNC(c3ccnc(CO)c3)=O)nn2)c(F)c1 Cc1cccc(C)c1OCC(N1CC2CC1CN2C(c1ccncc1Cl)=O)=O N1(C(C(=O)NC2COC2)C2CC2Cl)CCC(CO)C(NC(c2ccccc2)=O)C1 C12(NC(=O)C(O)CC(F)(F)F)CCCC1CN(C(c1cscc1Cl)=O)C2 C1(CNC(c2cnc(-c3cn(C)nc3)s2)=O)CCCN(C(c2ccn(C)n2)=O)C1 C(=O)(C1=CS(=O)CCC1)NC1C2CCN(C(c3cc(C)cc(C)n3)=O)C21 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(F)(C(=O)NC2CN(C3CC3)C2)CC1 C1(CNC(c2c(CNC(c3n(C(C)C)ccn3)=O)cco2)=O)CC2(CCO1)CC2 C1(C(N2CC(O)(CNC(CN(C(C)C)C)=O)C2)=O)CCc2c[nH]nc2C1 N1(C(C(CC)N(C)C)=O)CC(C)C(N=c2[nH]c(Cl)nc(C(F)(F)F)c2F)C1 c1(NC(c2ncc(C)c(OCC)c2Cl)=O)cnc(=NC(CC)CC)[nH]c1 CC1(C(=O)NCC(C2CCCCC2)NC(c2cnc(C3CCC3)o2)=O)CC=CC1 c1(OC)ccc(C=CC(=O)NCC2(O)CN(C(C3CCCC3SC)=O)C2)cc1Cl Cn1cc([N+](=O)[O-])cc1C(=O)NCCC1(O)CN(c2cc(Cl)ncn2)C1 c1(C(=O)NC(C2CCN(C(C3(OC)CC3)=O)C2)C)cc(Br)c2occc2c1 C=CCCCCC(=O)NCC1CN(C(=O)Nc2cc(Cl)ccc2NS(C)(=O)=O)C1 C1(CNC(Cc2nc(C)c(C)s2)=O)CCC(C)N(C(c2cnc(S)[nH]2)=O)C1 COn1cnc(C)c1C(=O)NC(C1CN(C(=O)C(C)CN(C)C)CCO1)C N1(C(C(CC)OC)=O)CCC(C)(C)C1CNC(c1ccc(F)cc1C)=O Cc1cc(Cl)cc2[nH]c(C(=O)NC3CCN(C(C4CN(C)C4)=O)CC3CO)cc12 C1(C(=O)NCCN(C(CC2CC(OC)C2)=O)C2CC2)CCN(CC(F)(F)F)C1 N1(C(C(c2cscn2)N(C)C)=O)CCN(C(=O)CCC2CCCC2)C(C(F)F)C1 C1(NC(c2ncn(C(C)C)n2)=O)CC2C(NC(C3CC4CC4C3)=O)C2C1 N1(C(C2CC(C)N2C(c2sccc2Cl)=O)=O)CC2(CCCC2)C1 N1(C(C(=Cc2ccccn2)C)=O)CCC2CN(C(=O)C=CBr)C2C1 C1(CNC(C2CC(CC)C2)=O)CN(C(c2ccncc2C)=O)CC2(CCC2)O1 C1(NC(C2CCC(=C)CC2)=O)CCC(C)N(CC2CC2)C1 N1(C(C(CO)OC)=O)CCC(CCNC(=O)Cc2ncc(C)[nH]2)CC1 N1(C(c2c(Cl)cc(C)s2)=O)CCCC2(CC(NC(=O)C(=O)NCC(F)F)CO2)C1 C1(CNC(C(CN(C(c2c(C)cco2)=O)C)C)=O)COCC1(C)C CC1CCC(NC(=O)C=CC2CCC2)CN1C(=O)CN1CCC(C(F)(F)F)CC1 CC1CC2CC2CC1C(=O)NC1CC2CNCC12 n1(CC(=O)NC2C(C)CN(C(C3OCCCO3)=O)C2)ccc2ccccc2c1=O c1(C(CNC(=NCCOC)N(C)Cc2nccs2)OC)c[nH]c2ccc(C)cc12 n1(C(C)C)ccc(=NC(=O)CC2CN(C(=O)CC3CCCOC3)CCO2)[nH]1 C1(CNC(C2(C)CC2)=O)CCCN1C(c1c[nH]nc1C1CC1)=O.c1(CO)ccccc1 N1(C(C=NOC)=O)CCC(C(=O)NCc2cncc(Cl)c2)C12CC2 C1(CN2CC(C)OC(c3ccccc3)C2)C2C3CC4C1C1C2CC3C41 N1(C(C(C(C)O)(F)F)=O)CC(O)(C2(CNC(c3nocc3Br)=O)CC2)C1 n1(CC)cc(C(=O)NC(c2cncs2)C)c(C)n1 N1(C(COC(N(C)C)=O)=O)CCC2CN(S(C)(=O)=O)CC12 C1(C(=O)NC(c2ccccc2Br)C(=O)OC)CCn2nccc2C1 Cc1c(C(=O)NCC(C)(O)CNC(C2COC2)=O)cnn1C C(N=c1[nH]ccn2nnnc12)C1(NC(c2c(CSC)cccn2)=O)CCOCC1 N1(C(CCC)=O)CCC(C)(C)C1CNC(=O)C(C1CCOCC1)OCC C1(CN(C(CCNC(C2C(C(C)C)CCC2)=O)=O)C)CC2C=CC1C2 C#CC1CCC(CNC(C2CCC(CNC(C3(C)C=CCC3)=O)O2)=O)CC1 C1(C2CCN(C(c3ccccc3)=O)C2)(C(N2C3(CN(C)C3)CC2)=O)CC1 C1(CC)CN(C(c2cc(C(F)F)ccc2F)=O)CCC1NC(=O)C(CC)C(C)C C1(NC(CCOC)=O)C2CC1N(C(C1(Sc3ccc(NC(N)=O)cc3)CC1)=O)C2 N1(C(COCCC#C)=O)CC2CCC(C1)C(NC(c1sc(C)cc1Cl)=O)C2 C1(NC(C=Cc2c(C)ccs2)=O)CCC(C)N(C(=O)COc2ccc(F)cn2)C1 c1(C(=O)OCC)cc(Nc2occc2OC)cnc1OC.c12cncc(c1)NC2=O c1(C(N2CCOCC(NC(CCCCN(C)C)=O)C2)=O)cc2c(cc1O)OCO2 Cc1cccc([N+](=O)[O-])c1C(=O)NCC(CNC(=O)C1=CC(C)CC1)CO c1(C(N2CC(OCCNC(CCC=CCC=C)=O)C2)=O)cc2nccn2c(O)n1 N1(C(CCCC#C)=O)CCCC(O)(CNC(c2cc([N+](=O)[O-])oc2C)=O)CC1 N1(C(C(COCC)C)=O)CCCOC(CNC(=O)C(CO)OC)C1 C(=O)(C1=COCCO1)NCCC(C)(C)NC(c1cccc(N2CCOC2=O)c1)=O c1(-c2onc(CC(C(CC)C)O)n2)cc(C#N)ccc1C Cc1[nH]c2ccccc2c1S(=O)(=O)N(CCCCN1CCc2sccc2C1)CCO CC(C)(C)CCCCC(=O)NCC1OCCC1C(N1CC(n2cccn2)C1)=O c1(OC)ccc(C)cc1NC(=O)C1=NOC(CNC(=O)C(C)C2CC2)C1 C(c1cnc(O)nc1O)=CC(N1CCC(OCCNC(C(CC)(C)CC)=O)C1)=O c1(C(=O)NC2CC(n3cc(CCCNOC)nn3)C2)cc2ccc(SC)cc2[nH]1 C1(C(=O)NC(c2ccc(O)nc2)C)C2CCN(C(c3ccc[n+]([O-])c3)=O)CC12 c1(C(=O)NCC2N(C(C(C=C)O)=O)CCC(C)C2)c(C)ccc2nonc12 N1(C(CSC)=O)CCCOC2(COCCN(C(=O)Cn3nnnc3C)C2)C1 C1(CNC(CC(CC)SC)=O)CN(C(C2CCOC2)=O)C2CCCCC12 C1(NC(c2ccc(CC)cn2)=O)CC2CC1N(C(=O)CCCNS(C)(=O)=O)C2 CC(C(CCc1ccccc1)NC(C1(NC)CC1)=O)NC(c1cnc(C#N)s1)=O c1(CCC)ncc(C(=O)N(CCCNC(C2(C3CC3)CC2)=O)CC)s1 C(=O)(C1=Cc2ccccc2C1)NCC1(O)CCN(C(C2OCCN(C)C2=O)=O)C1 N1(C(C(CSC)(C)NC(=O)CC2CC=CCC2)=O)CCC2(C=CCO2)C1 CC(C)C(C)(CO)NC(=O)CC=CCNC(=O)CCCNC(N)=O C1(CNC(C(C2CN(C(c3cn(C)nn3)=O)C2)OC)=O)CC12CCOCC2 c1(N(C(=O)N(CC(=O)NC)C2CC2)C)ncnc2scc(-c3cccs3)c12 c1(C(=O)NCC2C(NC(=O)C=CCO)CCC2)c(O)cc(O)cc1O c1(C(N2CCC(=O)C2c2cccnc2)=O)ccn2ccsc12 N1(C(C(CC)NCC)=O)CCN(C(=O)C=CC(=O)N(C)C)CC1CF.C(C)(=O)OC N1(C(CCc2onc(C)n2)=O)CCN(C(=O)CC(C)O)CC1C1CC1 C1(NC(C2C(CC)CCCC2)=O)CN(C(=O)CC2CSC2)CC12CCCC2 c1(Cn2c(-c3ccc(C)[nH]3)nc(CCCC)n2)cc(F)cc(Cl)c1 c1(C(=O)NCCOC2CN(C(C(C(C)(C)C)SC)=O)C2)cc(C)cc2c1OCC2 c1(C(N(CC(CNC(c2c(C)cco2)=O)(C)C)C)=O)cc(N)c(F)cc1C Cc1cn2ccc(C(=O)NC3CC4CN(C(C5CCCC5(F)F)=O)CC34)cc2n1 C1(OCCNC(C2C(C=C)C2)=O)CCN(C(C2CCOC2)=O)CC1 N1(c2ncc(C)c(CO)n2)CCN(C(=O)C=CCNC(=O)C(C)(C)C)CC(O)C1 c1(CC=C)ccccc1C(=O)NCC1(F)CN(C(C2C3CCC2CC3)=O)C1 C1(NC(C(C)NC(CC)=O)=O)CCC(NC(=O)C(C)(C)n2cccn2)C1 CCCCCCCS(=O)(=O)NC(=O)Cc1ccc(-c2cnn(C)c2)cc1 C1(NC(c2c(C)snn2)=O)CC2CC(NC(=O)CCC3CCC(=O)NC3)CC2C1 C1(C(N(CCC(=O)N(C)Cc2cc(C)nn2C)C2CC2)=O)CCOCC1(C)C c1(NCCCCC)cc(S(=O)(=O)NCC(N2CC3CCCC23)=O)ccc1Cl Cc1nc2cccc(C(N3C4CCC(C4)C3CNC(c3nnn(C)n3)=O)=O)c2[nH]1 CC1CCn2cc(C(=O)NC3CC4CC(NC(=O)CCN5CCC5)C3C4)nc2C1 C(CCC(=O)NCC1CCCC1NC(c1ccnn1CC(F)F)=O)OCC C=C1CCC(C(=O)NCCCC2CCCN2Cc2nc(C)c(CC)o2)CC1 N1(C(C(=O)NCCOC)=O)CCCC(N(C)C(c2ccncc2O)=O)C1 C(CCC)(C(O)C(=O)N1CCCc2nncn21)NC(C(CCCCCC)(C)C)=O CC1CCc2sc(C(=O)OCC3OCCC3F)cc2C1 N1(C(C2C(C(=O)OCC)C2)=O)CCCC(NC(c2conc2C)=O)CC1 C(=O)(C=CS(C)=O)NC1(C2N(C(COc3cc(C)on3)=O)CCC2)CC1 C(CC(C(=O)N1CCC(C(C)OC)CC1)NC(=O)CNc1ncccn1)=CC C=C(C)CC(C(=O)N1CCC(C(=O)NC2CN(C)CC2(F)F)C1CC)OC c1(C2CN(C(=O)NCc3nc(C)c(Br)s3)C2)ccc2ncsc2c1 c1(C(=O)Nc2c(OC)nccn2)cc(NC(C2CC2C(=O)NC)=O)cc(C#N)c1 c1(OC)ccc(F)cc1CC(=O)N(C1CCCCC1NC(=O)Cc1cnns1)C CCC(CC)CCCC(=O)NCC1(C(=O)NCCC2CC(C)(C)CO2)CCCC1 C(=O)(C1=CCCOC1)NCCCOCCNC(C1C(C)OC(C)C1)=O Nc1cc(C(=O)NC2CN(C(c3c[nH]c(=O)cn3)=O)CC3CC23)ccc1Cl c1(C(=O)NC2CCC(CNC(C3C(C)C3C)=O)C2)cncc2ncn(C)c12 N1(C(c2cc(CC)n(C)n2)=O)CCC(C2CCN(C(c3ncccc3C)=O)C2)C1 c1(C(=O)NC2CCCCCN(C(C3C=CCC3)=O)C2)ccc2ccc(O)nc2n1 N1(C(CN(C)CC)=O)Cc2nccn2CC(NC(=O)CNS(C)(=O)=O)C1 N1(C(CC(=C)C)=O)CC(NC(=O)C(C2CCCO2)C2CC2)Cc2ccccc21 c1(CNC(C2CCCO2)CC)cc(Br)cc(C)n1 c1(CCC)noc2nc(C)cc(C(N3CCC(O)(CN(C)C(C)=O)C3)=O)c12 Cc1[nH]nc2ccc(C(=O)NCC3C(C)CCCN3C(=O)COCCF)cc12 c1(C(C)C)nc(=NC(CNC(=O)CC(c2ccccc2)C2CC2)C2CC2)s[nH]1 c1(C(=O)NCC2(F)CN(C(c3ccc(F)cc3F)=O)C2)cc2n(n1)CC(F)C2 c1(CC(N2CC(SC)C(NC(=O)CCCC(C)(F)F)C2)=O)ccc2[nH]ccc2c1 C1(CC(=O)NC2CC(C)C2O)(NC(Cc2nc(C)[nH]n2)=O)CCCCC1 c1(CCC(=O)NCC2C(NC(CCCC#C)=O)CCC2)cccc(F)c1Cl c1(C(N(CCCCNC(=O)CC2CC2)C)=O)cc2c(o1)CCCC2 c1(OC)cnc(Br)c(NC(C2(C)CCCN(c3ccnc(C)n3)C2)=O)c1 c1(C(N2CC(C)C(NC(=O)CC3CC(=O)NC3=O)C2)=O)cc2cnn(C)c2s1 CC1=NOC(C(=O)NC2CCN(C(c3cn(C(F)(F)CO)nn3)=O)C2)C1C c1(CN(C)C(c2cnns2)=O)ccccc1CNC(c1cccs1)=O Cn1ncc2cccc(COC(c3cccc(-c4ccc(Cl)cc4)c3)=O)c12 c1(C(N(C)CC2CCCN2C(C2COC(=O)N2)=O)=O)cc2cc(Cl)sc2[nH]1 C(c1nc2ccccc2[nH]1)=CC(=O)NCCC(C)(C)NC(C(C1CC1)OCC)=O c1(C(N(CC(CN(C(=O)CC2CC23CC3)C)O)C)=O)cnnc(O)c1 N1(C(COCC(=O)NC)=O)CCC(NC(C2(F)CC2(F)F)=O)C1 c1(NC(C2CNCCC23CCC3)=O)cnc2ccc(F)cc2c1 Cc1cccc2cc(C(=O)NC(CNC(=O)CN3CCC(C)C3)C3CC3)cnc12 CC1COCCC1C(=O)NCC12CC1CN(C(C1(OC(C)C)CCC1)=O)C2 c1(C(N)=O)ccc(C(=O)NC2CCOCC2NC(=O)Cn2nnc(=O)[nH]2)cn1 c1(C(N2CCC3(CC2)CC(F)C3)=O)cn2c(n1)CCN(Cc1cn[nH]c1)CC2 n1(CC)cccc1C(N1CCCC1CN(C(c1cncnc1)=O)C1CC1)=O CC1(CNC(C2CCCN2C2CCCC2)=O)CCN(c2nnc(C(F)F)o2)C1 O=C(C1=CCCC1)NC(C(=O)NCCC1CCCC2CC12)C1CCC1 N1(C(C(N2CCCC(O)C2)C)=O)CCCC2(CCCN2C(=O)C2=CCC2)C1 C1(N)(C(=O)Nc2cc(C)n(CC3CC3)c2C)CC2CCC(C2)C1 CC1CCCC(c2nnnn2CCCF)(NCCCc2cnn(C)n2)CC1 N1(C(c2ccc(C(C)=O)s2)=O)CC(C2(NC(=O)CCCC(=O)N(C)C)CC2)C1 c1(-n2c(-c3cc(O)nc(O)n3)nc(CC(C)OC)n2)cc(C)ccc1C C1(S(C)(=O)=O)(CNC(C2(Cl)CC2C(N2CCC(C(=O)OCC)C2)=O)=O)CC1 C(CCCCCCCO)=CC(=O)NCC(=C)CCNC(c1occc1C)=O c1(C(=O)OCc2cccc(C(C)=O)c2C)cc2c(Br)cc(C)cc2[nH]1 C(C)(C)(CCCNC(C1CC12CC2(F)F)=O)NC(CN(C)C(N)=O)=O C(=O)(C#CC1CCCOC1)NC1CCN(C(C2(N(C)C)CCCC2)=O)CC1O C1(CNC(C(CCC2CCCC2)NC(=O)CC23CCCC2C3)=O)CC2CCCC2C1 C1(C(N(C(C)C)CCNC(=O)CN(C)CCO)=O)OC(C)(C)OC1(C)C C(=O)(C(CCOC)OC)N1CCC(NC(c2cc(COC)no2)=O)C1 c1(C(=O)NC2CC(NC(CC(C)C(F)F)=O)C(O)C2)cc2ccc(Cl)nc2s1 C(CC(C(=O)NC)NC(=O)CN(CC(=O)NCCc1scnc1C)C)OCC N1(C(C2CCC(C(=O)OC)C2)=O)CC=CC(NC(=O)CO[Si](C)(C)C)C1 c1(NC2CC(C)N(C(c3cc[nH]n3)=O)C2)ncn(C)c(=O)c1Br C1(NC(c2n(C)cnc2)=O)CN(Cc2ccc(Cl)c(Cl)c2F)CCC1(F)F c1(N(C)CC)nc(=NCCSC2=NOC(C)(C)C2)[nH]c2cc(C(F)(F)F)ccc12 N1(C(CC2(C)CCC2)=O)CCC(F)CC1C(N1CCC(CN(C)C)C1)=O N1(CC(c2ccccc2)=O)CCc2cccc3c2C(CCC3)C1 c1(CC)nc(Cl)nc(NC2CN(C(=O)C(C)OCc3ccncc3)CC2C)c1Cl c1(CC(=O)NC2C(NC(C(CC)(C)OC)=O)CCCC2)c[nH]c2ncccc12 c1(C(=O)NC(C(C(C)C)NC(=O)Cn2ccnn2)C)ncc(Br)cc1O N1(C(C2C3CC4C(C3NC(C35CCN(CC3)C5)=O)C24)=O)CC2C3C=CC(O3)C2C1 c1(C(=O)NCCCNC(=O)OC(C)C)cccc(C(C)(C)O)c1 Cc1ccc(C)c(C(=O)NC(C)C(N2CCCC(CO)C2C)=O)c1 N1(CC)CCC(CNC(=O)C(C)(C)CNC(C2C=CCC2)=O)CC1 CC1CCC(C)(C(=O)N(C)Cc2ccc(CNC(c3coc(C#N)c3)=O)cc2)C1 C1(C(N2CC(C)C2C(=O)N(C2CCCCC2)CCO)=O)CCOC(=O)CC1 N1(C(C(C)N(C)C)=O)CC(C(F)(F)F)C(CNC(C23CC(C#N)(C2)C3)=O)C1 C1(CNC(CN(C(COC)=O)C)=O)CN(C(=O)CC2(C#N)CC2)CCC1C Cc1nccn1C(C)C(=O)NC(c1cn(C)nn1)C(=O)N(C1(CCO)CC1)C C12(C(=O)NC(CN(C(c3c(C)nc(N(C)C)s3)=O)C)C)CCCC1C2(F)F C(CCC1CC1)(C(=O)NC1CCCC(=O)N1)NC(CC(C)SC)=O CC1CCC(C)N1CC(=O)NCc1ccc(CNC(=O)C2=NOCC2)cc1 c1(CC(=O)NC2CCN(C(c3csc(CO)n3)=O)C2)cccc(-c2cn[nH]c2)c1 N1(CC)CCOC(C(=O)NC(CC2CC2)CC(=O)NC(c2ccccn2)C)C1 C(=O)(CCC(=O)NN(C)C)N1C2CC(C(N(C)Cc3c(C)n(C)nc3)=O)C1CC2 N1(C(C(CC=C)CC=C)=O)CC(C)OC2(CCN(C(C3COC(=O)C3)=O)CC2)C1 c1(C(=O)NCC2OCCN(C(C(C(C)(C)F)(C)F)=O)C2)c(Cl)oc2ccccc12 C(C(C(=O)N1CCCCC1CCO)C(C)C)NC(c1c(C)c[nH]c1)=O c1(COC)ccccc1CC(N1CCCCC1C1CCN(C(=O)CC2CC2)C1)=O C#CCCN=C(NCCCn1cccc1)NCc1ncn(-c2ccccc2)n1 CC(C)C(C)C(CNC(c1csc(S)n1)=O)NC(c1csnn1)=O CC(C)CCCCC(=O)NCC#CC(=O)NCCN1CCOC1=O c1(OC)ccc(I)c(C(N2CC(OC)CC2C(=O)Nc2ccc(C)c(F)c2)=O)c1 C(C1=NOC2CN(C(=O)CC(C)(C)CCOC)CC12)NC(c1ccc(CC)[nH]1)=O c1(OC)cc(C=CC(=O)NCCNC(=O)CN2CC(C)(C)C2)cc(Cl)c1OC c1(CC(C)NC(=O)C(=O)NC2CNC(=O)C2)c(F)cc(Br)cc1F N1(CC(=O)N(CCCn2cc(C3(n4ccnn4)CC3)nn2)C)C(=O)CNC1=O Cc1onc(C(=O)N(CCCNC(=O)CCN2CCCC2=O)C)c1Br C(=O)(CCCC(=O)NC1CCN(C(=O)C=CCF)C12CC2)NCC C1(NC(c2sccc2-n2cccc2)=O)CCCCCN(C(C2CC2C2CC2)=O)C1 N1(C(C(C)N(C)C)=O)CC(C(=O)O)CCC1=O.CCS(=O)(=O)Cc1cn(CO)nn1 c1(C(N(CCCN(C)C(c2c[nH]c(C#N)c2)=O)C)=O)ccccc1OCC(N)=O Nc1cc(C(=O)NCC(CO)NC(=O)CCC=CC(=O)O)ccc1-n1ccnc1 C1(CNC(c2c(CC)n(CC)nc2)c2nnnn2C)CCCCC2(C1)OCCO2 C=C(Cl)C(C)(C)C(=O)N1CC2C(CNC(=O)CN(CC(=O)NC)C)C2C1 C1(NC(C(CC=CCC)C)=O)CN(C(=O)Cc2ccccc2Cl)CC1(C)C N1(C(c2c(C)ccnc2O)=O)CC2(COC(CNC(=O)Cc3ccsc3)C2)C1 C1(CC(=O)NC2C(NC(=O)OC)C2)(C(=O)OC(=O)C(C)C)CCCC1.C(C)(C)(C)O Cc1cccc2c1CC(C(=O)NC(C)(CNC(=O)CC1CC1)C1CC1)O2 C1(NC(COCCOCC#C)=O)CN(C(=O)C=Cc2ccccn2)CC1N=[N+]=[N-] C(CCO)(C(=O)NCc1ncoc1CCNC(C1CC2C=CC1O2)=O)N(C)C c1(C(N2CCC(CNC(C(C)OC)=O)(CO)CC2)=O)ccc(N)c(Cl)c1O C=CC(C)(O)CC(=O)NCCc1ocnc1CNC(c1cc(O)nc(C2CC2)n1)=O N1(C(C2(C)ON=C(C)C2)=O)CC2CN(C(c3cc(CN(C)C)on3)=O)CC2C1 c1(N2CCN(CCOC)CC2)nc(=NCCS(=O)CC)[nH]c2c(F)cccc12 C(=O)(CS(=O)C(F)(F)F)N(C1CCCN(C(C#CC(=O)N(C)C)=O)C1)C CC(C)C(CNC(C1CCC(O)C1)=O)C(=O)NCCc1cncs1 C1(C(=O)NCCCOC2CCN(C(c3cc(C)[nH]n3)=O)CC2)(CC)CCCC1O N#Cc1ccc(O)c(NC(C2CCCC(NC(=O)C=Cc3ccncc3)C2)=O)c1 c1(C(=O)NCC(CCOC)NC(CN(C2CC2)CC)=O)ccnc(O)c1 CN=c1[nH]c(=NCCCCC#N)[nH]c(=NC2CCC(OC)C2)[nH]1 Cc1nc(C(c2nnnn2C2CC2)NCC(C)Cn2ccccc2=O)sc1C Cc1cccc(C(=O)NCCCC(C)NC(=O)CC2CCCCC2O)c1F c1(CC(=O)NCC(CC)NC(c2cccc(NS(C)(=O)=O)c2)=O)ccncc1Cl N1(C(c2ccc(CC)cn2)=O)CCC2(NC(c3cnc(Cl)[nH]3)=O)CCCCCC12 C1(C(N2C(CCCC)CCC2)=O)CC(F)CCN1C(=O)COCC c1(C(=O)NC2C3(CC(NC(COCCCOC)=O)C3)C2)cnc2nccnc2c1 N1(C(C23N(C(CCOCCC)=O)CCC2CCC3)=O)CCOC2(CCCC2)C1 c1(OC)ccc(NC(=O)CC2CN(Cc3c(C)cccc3C)CCO2)c(OC)c1 C12(C(N3CC(NC(=O)CCc4ccncn4)C(F)C3)=O)C3CC(CC13)C2(F)F C1(CNC(Cc2n(C(C)C)cnn2)=O)(CO)CCN(C(=O)C(F)C(C)(F)F)CC1 CN1CCC(C(=O)NCC2CN(C(=O)Cc3csc(-c4ncccn4)n3)C2)C1 c1(CC(=O)NC(CN(C(C2(C)C(C(=O)OC)C2)=O)C)C)cccc(C)c1F N1(C(CCOC)=O)CCN(C(=O)CCc2cc3ccccc3[nH]2)CC12CCC2 c1(C(N2CC(C)C(NC(c3cnc4nccn4c3)=O)C2)=O)nnn2ccccc12 C1(NC(c2nccc(C)c2)=O)CN(C(=O)C(C)OCOC)CCC1C(F)(F)F C1(CNC(CSCC)=O)CN(C(=O)C(C2CCC(=O)N2)C)CCC1(C)C C1(O)(CCC)CN(C(c2cc(CNC(C3CC3CC(C)C)=O)[nH]n2)=O)C1 C1(NC(C(C)=CC)=O)CC2(C1)CN(C(c1ccnn(C)c1=O)=O)C2 c1(C(=O)NCC(CN(C(C2C(C)(C(C)C)C2)=O)C)C)sc(C(C)(C)C)cc1N c1(C(N(CCCN(C(=O)CN(C)C2CC2)C)C)=O)ccc(-n2ccnc2)nc1 CC1ON=C(C(=O)N2CC(O)(CN(C(=O)CC3CC(F)C3)C)C2)C1C C1(CNC(c2c(C(C)C)occ2)=O)CCCC(NC(c2ccoc2C2CC2)=O)C1 N1(C(C2C(CC)OCC2)=O)C2CC=C(C(=O)N3CC4(CCC(C)OC4)C3)C1CC2 c1(C(=O)NC(c2ccncc2)C)cc(F)ncc1NC(c1cncnc1)=O C=CC1(C(N2CCCC2CNC(C2CCCC(C#N)C2)=O)=O)CCCCC1 Cc1nc(N2CCCC(c3nc[nH]n3)C2)c2c(C)csc2n1 C1(C(=O)NC(c2cnccn2)CC)(OC)CCCC(C)(C)C1 c1(C(N2CC3(CCN(C(c4c(C)nn[nH]4)=O)C3)C2)=O)cnn2c1NCC(C)C2 C1(C(=O)NCC2N(C(c3cnc(CC)s3)=O)CCOC2)CCc2c[nH]nc2C1 N1(C(C(C)=C2CCC2)=O)CC(NC(c2csc(-c3cnn(C)c3)n2)=O)CC(C)C1 N1(C(CCC(C)(C)C)=O)CCCCC12CCCN(C(=O)CCCn1ccnc1)C2 C1(C(=O)NCC(CN(C(=O)Cc2ccon2)C)O)CCn2c(O)nnc2C1 Cc1cc(O)c(C(=O)N(CCCN(C)C(c2cccc(C)n2)=O)C)nn1 C(=O)(C(CO)C(C)(C)C)N(C(CNC(c1c(C)c(C(F)(F)F)ccc1)=O)C)C C(=O)(CCC(CC)NC(c1cc(C)nc(O)n1)=O)N1CC(SCC)C1 CC1CCN(C(=O)C(c2cnccn2)C)CCN1C(C1CCCN1C)=O c1(C(N2CCCCC23CCSC3)C)nc2ccccc2n1Cc1nn[nH]n1 C1(CCNC(C2(CC)CCC2)=O)CN(C(c2ccc(F)c(Cl)c2)=O)CC(C)O1 c1(NC(CNC(n2cccn2)(C)C)=O)cn(C(C)(C)C)nn1 C1(C(=O)NC2(CNC(=O)C(c3ccn(C)n3)C)CC(OC)C2)CC2(CCCO2)C1 C1(CC)CCN(C(=O)C(CC(C)C)N2CCCCCC2)C(CC)C1 CCCC(C(=O)OC)NC(=O)CC1CCN(C(=O)CNc2ccc(F)cc2)CC1 C#CCCCC(C)C(=O)N1CC2CC1CN2CC(=O)NCC(C)C O=C1CCC(C(=O)N2CCC3(CC2)CN(C(c2ccc(Cl)o2)=O)C3)n2cccc21 c1(OC)ccc(NC(C2CC2CNC(=O)C(O)C(C)C)=O)c(O)c1 Cc1ccc2c(c1)CC(C(=O)NCCCN(C(=O)Cc1ccoc1C)C)S2(=O)=O c1(C(N2CC(CCCC)N(C(c3sccc3C)=O)CC2)=O)ccc(F)c(F)c1C Cn1cnnc1CCCNC(C(C)(C)C)c1nnnn1Cc1ccccc1 N1(C(c2ccc(C(C)(C)C)s2)C(=O)NC)CC2(CCCCC2)C1 N1(C(Cc2ccc(C)s2)=O)CCC2CN(C(C3CC3(Cl)Cl)=O)CC2C1 S(=O)(=O)(c1cc(Br)ccc1Br)N1C(C(=O)NCCc2ccc(O)cc2)CC(=C)C1 c1(C(=O)NCC(C)(C2CCC2)NC(C(C)C#N)=O)cccc(CS(N)(=O)=O)c1 C12(NC(=O)CCOCCO)CCC(CC1n1cc(CO)nn1)C2.c1cccc(Cl)c1 C1(CC)CN(C(=O)CCC)CC1NC(=O)CCN(C)CCO N=c1[nH]cc(C(N2CCC(C(F)C(=O)NCCN3CCC3)C2)=O)o1 C1(OC)(CNC(=O)CCc2conc2C)CCN(C(c2csc(CO)n2)=O)C1 c1(OCC)cccc(CNC(=O)NC2CNC2)c1.c1(C(F)(F)F)ccc(OC)nc1 CCCCC(C(=O)NCC(C)N(C)C(C1CCC(=O)N1)=O)C(C)C C1(CC)CN(C(=O)C#CC(C)C)CCC1CNC(C1CCCN(CC)C1)=O C#Cc1cccc(N(C(=O)C(C2CC2)N(C(=O)Cn2cncn2)C)C)c1 N12CCN(CC1)C2CNC(=O)C1CC1.c1(CC(=O)OC(C)(C)C)cccc(F)c1 C(=O)(CCCC(C)=O)N(CC(CNC(C1(NC(C)=O)CCC1)=O)(C)C)C N1(CC)CCCC(CNC(=O)C(C)(C)C2CCN(C(=O)CCc3ccco3)C2)C1 N1(C(C2COC2)=O)CCN(C(=O)C=CC2CCCO2)CC(CO)C1 CC1c2ccccc2CCN1C(c1cc2c(s1)CCN(C(C1CCCO1)=O)C2)=O C1(S(C)(=O)=O)(C(N(CC(C)CNC(=O)C(C)(C)C2CCCO2)C)=O)CCCC1 c1(C(N2CCC(CNC(c3cc(CC)no3)=O)(OC)C2)=O)cccc2nc(O)oc12 C1(C(N2CC(O)(CCC)C2)=O)CCC(C)N(C(C2CCCC(C)CC2)=O)C1 N1(C(CC2CCCN(C(Cc3onc(C)n3)=O)C2)=O)CCC(F)C(F)C1 CC1(C)CN(C(c2cc(O)cc(O)n2)=O)CC1NC(=O)CCC(N)=O CC1CCCC1(C)C(=O)NCCN(C(c1cncnc1C1CC1)=O)C1CC1 N1(C(CNC(CC)=O)=O)CC2(CCN(C(c3c[nH]ccc3=O)=O)CC2)C1C(C)C c1(C(=O)NC2CN(C(c3ccc(NC)cc3)=O)CC23CC3)cc(F)c(Cl)cc1F CC1CN(C(c2cncc(N)n2)=O)C(C)CN1C(=O)CCc1cccnc1 c1(C(=O)NCC(CNC(=O)CC2OCCC2(C)C)OC)cnc2cc(C)nn2c1 CC(C)(CC(=O)NC1CCCCCC1NC(=O)CSc1cccc(F)c1)C(F)F c1(C(=O)NC2CC(CC(=O)NC(CC=C)CO)C2(C)C)cc2n(n1)CCO2 N1(C(C2(c3ccccc3)C(C)(C)C2)=O)CCCC(NC(C2CCCCS2)=O)CC1 c1(OCNC(=O)C=C2CCC2)csc(C2CCCN2CC(F)F)n1.O=CO C1(CNC(C2CC(CC)(CC)C2)=O)CCCN(C(C2CC(=C(F)F)C2)=O)C1 c1(C(N(CC(C)NC(C2(Oc3ccccc3)CC2)=O)C)=O)ncn2ccccc12 c1(C(=O)NC2CN(C(Cc3nnc(C)o3)=O)C3C2C3)c(F)cncc1Cl Cc1nc(C(=O)NCC2(NC(=O)CN3CCC(C)C3)CCC2)c2n1CCCC2 Cc1nc2ccc(C(N3CC(O)C(O)C3CNC(C3CC3(F)F)=O)=O)cc2[nH]1 N1(C(CCCOCCC)=O)CC(O)(C2CCN(C(=O)C(C)CC(F)(F)F)CC2)C1 c1(C(N2CC(NC(c3n(C)ccc3)=O)C(C)(C)C2)=O)ccc(Cl)c(F)c1O c1(C(=O)OC)cc(C(=O)NC2CC(NC(=O)CC=C(Cl)Cl)C(O)C2)ccn1 C#Cc1cc(C(N2Cc3[nH]nc(C(=O)NCCCCOC)c3C2)=O)ccc1C CCCC(C)(C)CN=c1[nH]c(N2CCC3C(CCN3C3CC3)C2)nc2c1COC2 N1(C(C(COCC)C)=O)CC2(COC(CNC(=O)COC3CCC(C)CC3)C2)C1 C12(C(=O)NCC3C(CNC(C(CC)=CC)=O)C3)CCC(CC1)C2 c1(C(=O)NCC2CN(C(CCCCCNC(N)=O)=O)C2)c(F)cc(F)cc1Cl N1(C(c2c(C)ncs2)=O)CC(NC(C2(C#N)CCCCC2)=O)CC12CCCOC2 C1(NC(=O)CSCc2ncc[nH]2)CCCN(CCCNC(C2CC2F)=O)C1 CC1(C)CCCCC1=CC(=O)NC1CCCC(NC(C2CC(F)(F)C2)=O)C1 C1(C(=O)NCC2CC=CCC2)N(C(=O)CCc2ccco2)CC12CCCC2 CN1CCCC1C(N1CC(O)(CCNC(C2(C(F)(F)F)CC(O)C2)=O)C1)=O c1(COC)ccc(C(N2CCOCC2CNC(C2CC2c2nc[nH]n2)=O)=O)cc1 C=C(C)C(C)(C)C(=O)NC(C)CN(C)C(C1CSCN1C(c1cccs1)=O)=O C1(OC)CCCC(C(N2CCN(CCNC(c3cc(C)[nH]c3C)=O)CC2)=O)C1 C1(CC(=O)N(CCCCCC=C)C)C2CCC(C2)N1C(C1CC(C)N(C)C1)=O C1(C)(C(N(C)CC2(O)CCN(C(=O)CCS(N)(=O)=O)C2)=O)CC2CCC(C1)S2 CCC(C)CCC(=O)NCCC(C)N(C(=O)CC(C)(C)O)C C1(C(=O)NC2CCN(C(c3cnn(C(C)C)c3N)=O)C2)CCCC2(C1)CC2(F)F N1(C(C(C)NC(COC)=O)=O)CCC(NC(C2CC(C)(C)C2)=O)CC1C C1(CNC(=O)CSC2CC2)(CO)CCCN(C(C2CC3CCC3C2)=O)C1 CC(CC1CCC1)C(=O)N1CCCC1C(C)(C)C.c12cc(on1)CNC(=O)CO2 c1(SC)ccc(C(=O)N(C)CCN(C(=O)CCOCC2CC2)C)s1 CC(C)C(F)(CNC(=O)CC(C)C(F)F)C(=O)NCCN(C)C(=O)C1CC1 C1(NC(CC2CC(=O)NC2)=O)COC2C(NC(c3cn(C(F)F)cn3)=O)COC12 C1(C(=O)NC2CN(C(C3N(N=O)CCCC3)=O)C2)CC2COCC(C1)C2 S(=O)(=O)(c1cnc(N(C)Cc2ncc(C(C)C)o2)cc1C)N1CC(Br)=C(C)CC1 C=CC1(CC(N2CCC23CN(C(c2ccc(C4CC4)cn2)=O)C3)=O)CCOCC1 Cc1cc(-c2noc(CC3(C)COCCO3)n2)cc(O)c1 CC1C(NC(C2CCCC(O)C2)=O)CC2CCC1N2C(=O)C(F)(F)C(O)C(C)C N=c1cc(C(=O)NC23CC(NC(=O)COc4cnc(Cl)cn4)(C2)C3)nc(Cl)[nH]1 c1(C(N2CCC(CNC(C(C)NC(C)=O)=O)C2)=O)ccc(Br)c(Cl)n1 C#CCCC(O)CCNC(=O)C(C1CN(C(c2cccc(O)c2C)=O)C1)OC Cc1cc(N)c(C)nc1C(=O)NCC1COCCN(C(C2CCCC(C)C2)=O)C1 CCS(=O)(=O)CC(=O)N1CCC(O)C(C(=O)Nc2ccc(N3CCCC3)nc2)C1 N1(C(c2c(C)cccc2)=O)C(C(=O)Nc2cnc3[nH]cnc3c2)CC2CCCC12 c1(C(N2CCN(C(c3cc(OC)ncn3)=O)CC2C)=O)ccc2c(c1)C(=O)NC2 Cc1cc(-c2nc(CCn3ccnc3)nn2C2CCC2)nc(C(F)F)n1 C1(CC(c2n(CCCSC)nnn2)NCCO)CCN(C(=O)CC(C)F)CC1 N1(C(=O)NCC2CCCCC2C(=O)O)CCC12CCCOCC2.c12ncc(s1)C2 C1(NC(C(C)OCC#C)=O)CN(C(C2(C)CC2)=O)CC1O N1(C(COC(CC)C)=O)CCC2(CCC(NC(=O)C3CCN(C)CC3)CC2)C1 CCC(C(=O)NCC1CN(C)CCN1C(=O)CC12CCC(CC1)CC2)C(C)O c1(N(CCCSc2ccccc2)CC)nc(N(C)C)nc2ccccc12 Cc1cc(C(=O)NCCCN(C(C2(CC3CCCO3)CC2)=O)C(C)C)cc(F)c1 c1(C(=O)NC2CC2CNC(c2cn(C3COC3)nn2)=O)cc2c(o1)CCCC2 c1(CC)ccc(O)c(C(=O)NC2CCCC2NC(=O)CCOCC(F)F)c1 C(N=c1[nH]c2c(F)cccc2o1)C1CCCC(NC(c2ccn(C)c2)=O)C1 C(=O)(CC(C)C1CC1)NCCC(C)N(C)C(c1ccco1)=O Cc1ccccc1C(C)NC(=O)CC1C2CN(C(C3CCSC3)=O)CC12 CN1CCC(C(=O)NC2CC(CCNC(=O)CS(N)(=O)=O)C2)CC1 N1(C(C(C(CC)C)O)=O)CC2CC(NC(c3ccnc(S)c3)=O)CC(C2)C1 N1(CCNCc2occ(C(=O)NCCO)n2)CCCCCC1 c1(OC)cccc(CNC2C=CC(C(=O)NCCOCCC(C)C)C2)c1C n1(CC(=O)N(CCCC(=O)NCc2n(CC)ccn2)C)cnc(C#N)n1 O=C(NNc1cccc(Cl)c1Br)NC1C2CCCCCC12 N1(C(c2cnc(SC)s2)=O)CCN(C(c2ccc(C)nc2N)=O)CC1CCO C1(OC)CN(C(=O)CC2COCCO2)CC1NC(=O)COc1cncc(F)n1 c1(CC)ncc(Cl)c(C(=O)NCCC2(NC(=O)CCc3ccc(Cl)cc3)CC2)n1 N1(C(CN2CC(=O)NCC2)=O)CC2(CC(C(=O)Nc3ccc4nccn4c3)CO2)C1 C1(NC(C=C(C)C2CCCCC2)=O)CCSC12CN(C(=O)C(C)(F)C(C)(C)F)C2 c1(C(N2CC(NC(C3CC(C(C)C)C3)=O)C2)=O)cnc(C(C)O)s1 n1(CC(N2CC(CCNC(CC3(CC)CCC3)=O)C2)=O)nnnc1C1CC1 C1(C(N2C(CNC(c3ccc(OC(F)F)nc3)=O)CC2)=O)CCCCCS1(=O)=O S(=O)(=O)(CC(=O)NCC1CC(NC(=O)CCCN2CCCC2)C1)NCC N1(C(C2(C#N)CC2)=O)CCCC12CCCN(C(c1cc(=O)n3ccsc3n1)=O)C2 C1(C(=O)NC2CCN(C(c3scc(OC)c3OC)=O)C2)CCn2c(C)cnc2C1 c1(C(=O)NCCC2C=CCC2)coc2c1CN(C(=O)Cn1ccnn1)C2 C#CCCCCC(=O)N1CC(O)(C(C)NC(=O)COC(F)(F)F)C1 C=CC(C)(C)C(=O)N(CC(C)NC(=O)Cn1nnc(-c2ccsc2)n1)C c1(NCC2CCC(NC(NOC)=O)C2)cnc(OC)nc1.C(C)(C)(C)OC(=O)N Cn1cncc1C(=O)NC1CCCC1CNC(=O)CCNC(=O)OC(C)(C)C C1(C(C)C)CN(C(=O)CN2CCN(C)C(=O)C2)CCN1C(=O)CN1CCCC1=O C1(C(=O)NCC2C(C)CCN(C(COC(C)C)=O)C2)CCc2nncn2CC1 C1(C)(C(N(C(C)CO)C)=O)CCCN1C(=O)Cn1cnnn1 C1(NC(c2snnc2C2CC2)=O)CCC2CC1CN2C(c1ccco1)=O N1(c2cc(OC)nc(C)n2)CC(NC(C2CC2(C)C(C)C)=O)CC2(CCC2)C1 c1(C(N2CCC(NC(C(CC=C)OC)=O)CC2)=O)c(F)cc(Cl)cc1F C(C(C)(C)CNC(=O)Cn1cnnn1)N(C(=O)COC(C)(C)C)C c1(C(N2CCCC(C)(C(=O)NC)C2)C(=O)NCCOCC)cc(Br)ccc1OC Cc1c(C(=O)NC2COCC2CNC(=O)C(C)SC(F)(F)F)cnc2ncnn12 C(=O)(C(C)N=c1ccn(CC(=O)NCc2ccc(Cl)c(Cl)c2)[nH]1)OCC c1(OC)ncc(Cl)cc1NC(c1cncc(NC(=O)CC#N)c1)=O c1(C(C(=O)NC2CC2CNC(c2snc(O)c2Cl)=O)=O)ccc2c(c1)CCC2 C(C)(c1ccccc1F)=CC(=O)NCC(C)N(C(c1c(SCC)cccc1)=O)C C1(NC(C(COCC)C)=O)CCC(NC)CC1.C12CN(CC1OC)C2=O C#Cc1ccc(NC(=O)CN2CCSCC2c2ccc(C)c(Br)c2)cc1 C1(C(N2CCC(O)(C(C)CNC(c3csnn3)=O)C2)=O)(OC)CCCCCCC1 c12nc(n(C)n1)C(=O)N2.C1(C(C)NC(COCC)=O)CN(C(=O)OC(C)(C)C)C1 C(=O)(CC(C)(C)C)N(CC(CC)NC(C1CC2C=CC1C2)=O)CC N1(C(CCCCSC)=O)CCCC(C)(NC(=O)CC2CCCOC2)C1 C(c1cc(Cl)c2c(c1)OCCO2)=CC(=O)NC1C=CCN(C(C(COC)O)=O)C1 CN1C(=O)CCCC1C(=O)N(c1cccc(F)c1)C c1(OC)c(CNC(=O)NCC2(C)NC(=O)NC2=O)ccnc1Cl Cc1c2c(-c3cnc(C(N4CC5CC5C4)=O)c(C(F)(F)F)c3)cccc2nn1C C1(CCC(=O)NCC(COC)O)CCCN(C(c2ccc(Cl)o2)=O)C1 c1(OCC)cc(C(=O)NC(C)(C(=O)NCC(C)N=[N+]=[N-])C2CCC2)on1 c1(C(=O)NCCOC2CCN(C(C3C(C)(C)C3(C)C)=O)C2)ccc2c(c1)CCO2 c1(CC(=O)NC2(CNC(C(CC)n3cncn3)=O)CC2)nc(C2CC2)nn1C CC(=Cn1ccnn1)C(=O)NCCCNC(c1cn(C)[nH]c1=N)=O C(=O)(C(C)CCC(C)(C)C)NC1CN(C(C(C)CF)=O)CC1(C)C C1(CNC(C(C)N(C)C)=O)N(C(c2csc(O)n2)=O)CCCC1(C)C C1(C(=O)NC2(CC=C)CCOC2)CCC(CNC(C2CCC2)=O)CC1 C1(NC(CS(C)(=O)=O)=O)COC2(C1)CN(C(c1ccc3c(c1)C=CC3)=O)C2 c1(C(=O)NCC2C(CNC(CC(C)c3cnn(C)c3)=O)C2)cc(C(F)F)nn1C c1(C(N2CCN(C(=O)C=Cc3ccccc3F)C3C2C3)=O)ccc2c(c1)NCC2 c1(OC)cc(C(=O)NCC(C)(C)C(=O)N(C)Cc2cn(C)nn2)ncn1 c1(C(=O)NCC2(C)CCN(C(CCC(=C)Cl)=O)C2)ccc(Cl)c(C#N)c1 c1(NC(C2CC(NS(=O)(=O)C(F)(F)F)C2)=O)cc(O)nc(O)n1 C1(CC=C)(C(=O)NC2CC2NC(c2csnc2Cl)=O)CCOCC1 N1(C(C(CCF)OC)=O)CCC(C(=O)N(CC2CCCCC2)OC)C1(C)C CC1CC(CNC(C2(F)CCCCC2)=O)CCN1C(=O)COCC1CCCCC1 C1(CNCC2CCC(C(N3CC(C)(C(N)=O)C3)=O)O2)CCC(F)(F)C1 c1(C(C(=O)NC2CCC2)N(CCN(C)C)C)c(Br)cnn1C c1(NC(=O)NC2C(OCC)COCC2)cc(CO)cc(C)c1 c1(CC)cccc(F)c1NC(=O)Nc1nc(N(CCCOC(C)(C)C)C)sn1 N1(C(C)=O)CCCC(CC(=O)NCCOCCN(C(=O)C(O)c2ccsc2)C)C1 N1(C(C2C=CC(n3cc(SC(C)C)nn3)C2)=O)CCOCC1c1cccc(F)c1 c1(OC)ccccc1CC(N1CCCC1=O)C.c1(CS(=O)(=O)NC)ccccc1C c1(C(N2CC(C)C(NC(C3CC3(Cl)Cl)=O)C2)=O)ccc2c(c1)CCCCC2=O CC(=O)CCCCC(=O)N1CCC(NC(=O)CC2CC2C(F)(F)F)CC1 Cc1nccn1C(C)C(=O)NCCC1(C(N2CC(CC(F)F)C2)=O)CC1 c1(C(=O)NC2CN(C(=O)C#CC3CC3)CC23CC3)cc(F)c2c(c1)CCC2 C1(C2(CNC(=O)NCc3nnc(C4(C)CCO4)o3)CC2)CCCCO1 c1(C(N(C)CCN(C)CC2(C)CC2C(=O)O)=O)cncc(C(=O)OC(C)(C)C)c1 N1(C(CC(CNC(c2cccc(C)c2N)=O)(C)C)=O)CCNC(=O)CC1C c1(OC)ccc(F)c(F)c1C(N1CCC(O)C1C(=O)Nc1ncc(C#N)cc1Br)=O c1(CC)ccccc1C(=O)N(CC(C)(C)NC(=O)CC1CC2(CC2)CO1)C N1(C(C(CCOC)NC(c2cc[nH]c(=N)n2)=O)=O)CC2CCOC2C1 C1(CNC(C2(COCC)CC2)=O)(CO)CC12CCN(C(=O)C(C)(F)F)CC2 CC(C)C(C)C(=O)N1CCC(OCCNC(c2cnc(S)nc2)=O)C1 N#Cc1cncc(CNc2nc(Cl)ccc2C(=O)NCCc2cccnc2)c1 c1(C(=O)NCC(C)(C)NC(CCC(=O)NCC)=O)ccc2nc(S)oc2c1 N1(C(CC2C(C)CCO2)=O)CC(CO)C2(C1)CN(C(C1(C)CCCO1)=O)C2 CN1CCC(C(=O)NC2(CCC(=O)NC(C)(CO)C3CCCC3)CCC2)CC1=O Cc1cnc(C(N2CCN(C(c3cc(C4CC4)no3)=O)C(C(C)C)C2)=O)c(F)c1 CC1CCCN(C(=O)C(F)=CCCF)C1CNC(=O)Cc1csc(C(C)(C)C)n1 c1(OC)cc(OC)cc(C(N2CCC(CNC(=O)CC(C)SC)C(C)C2)=O)c1 N1(c2ccnc(NCCN3C(=O)CCC3)n2)CCn2ncc([N+](=O)[O-])c2C1 C1(C(=O)NCCS(=O)CC)(NC(COCCCC)=O)CC(C)C1 c1(C(=O)NCCNC(c2n(C)nc(C3CC3CO)c2)=O)nc2n(c1Cl)CCCC2 N1(C(C(C)=C(C)C)=O)CC2(CCCN(C(=O)CC3CC(O)C3(C)C)C2)C1 C1(NC(c2nnnn2C)C(C2CCCC2)OCC)CNCC1C(F)(F)F C1(C(N2CC(N(C)C(c3ccc(O)nc3)=O)C2)=O)C2CCN(CC2)S1(=O)=O C1(NC(Cn2c(C)nnn2)=O)CCC2(CCCN(C(c3cn[nH]c3)=O)C2)C1 C(=O)(CCCCCCS(N)(=O)=O)N1CC(C)(N(C(C(C=CCCC)O)=O)CC)C1 CC(C#N)C(=O)N(CCN(C(C)CCO)C)CCCC(=O)NCc1ccccc1 C1(NC(C2(OC(C)C)CCC2)=O)CN(C(=O)CC2C=CCC2)C(C)(C)C1 C(c1ccc(F)cc1F)=CC(=O)NCC(C)N(C)C(c1n[nH]cc1[N+](=O)[O-])=O N1(C(c2c(C)cns2)=O)CC2(C)CN(C(c3coc(C(F)F)n3)=O)CC2(C)C1 C(=O)(C1COc2ccccc21)N1CCC(NC(C=COCC)=O)C2(C1)CCC2 C#Cc1cnc(C(=O)N(CCCN(C)C(c2ccc(N)cc2Cl)=O)C)c(C)c1 C1(CNC(COCCC=C)=O)CCC2(CCC2)C1NC(C1C2(CC2)C12CC2)=O c1(OCC)ccc(Cl)nc1C(=O)NC1CCN(C(=O)CCC2(C)CC2)C(C)C1 N1(C(CCC(=O)OC)=O)CCC2CCCC12CNC(c1cc2oc(C)cc2[nH]1)=O C=CC(CC)C(=O)NC1(C(=O)OC)CC1.C12CCCN1C(=O)C1CC21 C1(C(=O)NCc2scc(C)n2)C2CC3C(C2NC(=O)CN2CCSCC2)C13 C1(CCF)C(=O)N1.Cc1ncc(Cc2cn(SCC3CC3)nn2)s1.Cc1ccsc1 Cc1nc(N2CC3(CCCC3NC(c3c(C)n[nH]c3C)=O)C2)ccc1C#N c1(NC(N2C(CC(=O)Nc3cccc(C4CC4)c3)CCC2)=O)ccc(Cl)nc1Cl CC1(C)CN(C(=O)CCc2ccco2)CC1NC(=O)CC1CC2(CCO1)CC2 C1(n2cc(CNC(C3C=CCS3)=O)nn2)CCN(C(=O)C(F)c2cnc[nH]2)CC1 c1(CN2CC(C)(C(=O)NCc3ccc(C)nc3Cl)C2)c(O)cc(Cl)cc1Cl S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C)N1C(C)(C(N2CCn3c(nc(C)n3)C2)=O)CC1 CC1(C(N2CC(N3CCNCC3)C2)=O)CCN(C(=O)C(Cl)Cl)C1 CC(C)(C(=O)NC(=O)C(O)CCC(=O)O)S(=O)(=O)c1ccc(Br)cc1 C1(C(F)F)(CNC(c2n(CC)ccn2)=O)CCN(C(C2COCC2COC)=O)C1 Cc1ccc2c(C=CCNC(=O)Nc3cccc(NCCC4CC4)c3)c[nH]c2c1 C(=O)(C(CC(C)CC)NC(c1c[nH]c(=NC)o1)=O)Nc1cc(CC)cc(O)c1 C1(C(N2CC(C(C(=O)N(CC(O)CO)CC)O)C2)=O)CC(C)(F)C1 c1(C(=O)NCCCN(C(=O)CC(C2CC2)C2CC2)CC)nn(C)cc1S(N)(=O)=O C1(C)(NCCN(C)CC)CCCN(C(=O)CCc2ccc(C3CC3C)o2)C1 c1(C(=O)NCC(CNC(C2CC(CCC)C2)=O)(C)C)cc(Br)cc(C)c1C C(C(=O)NNc1ccccc1C(=O)O)(n1cc(Cn2c(C)ncc2)nn1)N(C)C N1(C(n2cc(CCCC)nn2)C(=O)NCC(C)C)CCOC(Cn2cccn2)C1 c1(C(N2C(CNC(C(C)SC)=O)CC2)=O)sc2nc(C)c(C)c(C)c2c1N c1(C(N2CC(CNC(c3ccc(CC)[nH]3)=O)C(C)C2)=O)cccc(Cl)c1NC N1(c2cc(C(=O)OC)nc(C)n2)CCCC2(NC(C3CCCN3C=O)=O)CC2C1 c1(OC)cc(C(N2CCC(C)C(C(=O)NCC3(C)COC3)C2)=O)cc(Br)c1Cl N1(C(C2(NC(C3C(C(C)C)OCC3)=O)CC(F)(F)C2)=O)CCCC(C)C1C C1(NC(C2CC(OC)C2)=O)CC2(C1)CC2NC(=O)Cc1ncncc1Cl C(CC(C)CCNC(=O)C(C)(C)n1ccnn1)NC(C(c1ccccc1)OC)=O C1(C(=O)NCc2cccc(C)c2)N(C(c2ncn(C)n2)=O)CCCC1(C)C c1(OC)nc(C)c(-c2cn(CC(C)NC(=O)CC3CCCC(OC)C3)nn2)s1 Cn1nnc2c(NC3(C)CN(C(=O)CC4(O)CCCCC4)C3)ncnc12 c1(C(=O)NC(C(C)(C)NC(c2cnc(OC)s2)=O)C)ccc2c(c1)CC(=O)N2 Cc1ccc(C(=O)NCC2CCC2NC(=O)C(=O)Cc2ccccc2F)c(C)c1 N1(C(c2cc(O)ccc2Br)=O)CCN(C(=O)C#CC2CC2)C2(CC2)C1 N1(C(C(C(C)O)(F)F)=O)CCOC2CN(C(=O)CC3=CCN(C)CC3)CC12 CC(C)C(C)C(=O)NC(c1nocc1C(N1CC([N+](=O)[O-])C1)=O)C C(=O)(C1CCc2ccccc21)NC1CN(C(C(CSC)(C)C)=O)CC(C)C1 N1(C(C2(NC(c3ccc(NC(C)=O)cc3)=O)CCC2)=O)CC(S(C)(=O)=O)C1 c1(CC(=O)N(OCC)CC2CCN(C(=O)C(F)(F)CC)C2)sc(C2CC2)nc1C C(CCC(C)C)(C(=O)N1CCCC1C(=O)Nc1cccc(I)c1)NC(C)=O c1(CNC(C(C)NC(c2c(CC)occ2C)=O)=O)cc(C)cnc1O c1(C(=O)NCC2CCN2C(=O)Cn2cc(C3CC3)cn2)ccc(F)cn1 C(CC(C)C(=O)NC(C)CCC(=O)NC1CCN(C(N)=O)C1)OC N1(C(c2c(C)scc2)=O)CC2COCC2C1.N12CCC(O)(C1)c1nc(no1)C2 C(C)(C(=O)C1(C(=O)OC(C)(C)C)C(C(N(CCNCC)C)=O)C1)SCCC C1(CC)CCCN(C(c2cc(Cl)n(C)n2)=O)C1C(=O)NCc1conc1C C1(NC(C(CC)C2CCOCC2)=O)C2CN(C(c3ccc(N(C)C)cc3)=O)CC12 C1(NC(Cc2ccn(CC)n2)=O)CCCN(C(=O)Cn2ncc(O)nc2=O)CC1 C(C)(C(C(=O)N1CCC2(CSC2)C1)C(C)C)NC(c1c(CCC)n[nH]c1)=O c1(CC(=O)N(CCCN(c2cccnc2)C)C)cnc2ccccc2c1 N1(C(C#CC(C)C)=O)CCC(CNC(C2C3CCCC23)=O)C12CCC2 C#CCC(C(=O)N1CC(O)CC1CC)NC(=O)CNC(c1ccco1)=O C=C(CNC(C1(CCN=[N+]=[N-])CC1)=O)CCNC(=O)CSC CS(=O)(=O)CCC(=O)N1CC=CC1(C)C(=O)NCC1(F)CC(O)C1 c1(OC(c2cc(C(=O)OCC)n(C)n2)=O)ccc(-c2cncnc2)cc1F Cc1cn2c(=O)c(C(=O)NC3CC(CNC(C4COC(C)C4)=O)C3)cnc2s1 C(C(=O)NCc1nocc1C(=O)NCCC(=O)N1CCCC1)(C(C)C)OCC c1(C(=O)NCC23C(CN(C(C4(C)CCCCO4)=O)C2)C3)cnc2[nH]cnc2c1 c1(NC(=O)NC2CN(C(C3CCN(C(C(C)(C)CC)=O)C3)=O)C2)cccc(F)c1O c1(C(=O)NCc2ccc(CNC(=O)CC3(O)CC3)cc2)cncc(Cl)c1Cl C1(OCC)CN(C(c2nnn(C)c2C(F)F)=O)CC1CNC(=O)CO c1(C(N(C)CC2N(C(C(C3CC3)SC)=O)CCC2)=O)ccc2c(c1)NC(=O)C2 C#Cc1cc(NC(=O)CCCN(C)C(C2CCCC2C)=O)ccc1C C(C)(C(=O)N1CC(CNC(=O)CN2CCOCC2=O)C(C)C1)(C(C)C)NC(C)=O c1(C(=O)NC(CNC(C(C(C)C)OCC)=O)C)cc(C(F)(F)F)ccc1N c1(NCc2cc(CC)no2)ccc(S(=O)(=O)N(C)Cc2ncccc2Cl)c(Br)c1 n1(CC)nncc1C(N1CCC1CNC(c1cnn[nH]1)=O)=O N1(C(c2c(CC)onc2C)=O)C2CCC1C(F)C(NC(=O)CC(C)C1CC1)C2 N1(C(C(C)=C(CC)C)=O)CCC(C)(C)C1CC(=O)NCC(C1CC1)SC c1(C(=O)NC2CN(C(c3ccc(C)n3C)=O)CC2O)cn2c(n1)CCC(C)C2 c1(C(=O)NC2CN(C(C3(OC)CCC3)=O)CC2C(F)F)sccc1S(N)(=O)=O C12(CNC(C(CC)Oc3ccccc3)=O)COC(CNC(C3CC(=O)N3)=O)(C1)C2 CC(CN(C)C)CC(=O)NCC1(O)CCOCC1.C1C(=O)N1 Cc1cc(O)ccc1NC(C1CCN(C(=O)Cc2cccs2)CCO1)=O Cc1cc(C(C)C)ccc1C(=O)NC1COCCN(C(C2C(C)C2C)=O)C1 N1(C(COc2ccc(C)cc2)=O)CCC2CC(NC(=O)CCCCO)CCC2C1 c1(OC)cccc(CNC(c2cn(C3CC(C)C3)nn2)=O)c1.C12(S)CCC(CC1)C2 c1(C(=O)NC(C)CNC(=O)C(F)C2CCOC2)ccnc(CN(C)C)c1 c1(CC(=O)NCC2CCN(C(C3C(CCC)C3)=O)C2)cccc2c1OCCO2 C(=O)(CC(O)C(C)C)NC(C(=O)NC(CC#C)(C)C)C(C)O Cc1cc(C(N2CC3CC2CN3C(C2(F)CC=CCC2)=O)=O)ccc1O C(=O)(C(C)n1cncn1)NCCCN(C(=O)Cn1ccnn1)C(C)C Cc1cccc(C(=O)Nc2csc(-c3ccc(SC(F)(F)F)cc3)n2)c1Cl c1(C(=O)NCc2ccc(C(=O)NOCC3CCCO3)s2)ccc2n[nH]cc2c1 Cc1noc(C)c1CCC(=O)NC(C1CCCN1C(=O)C=Cc1cnc[nH]1)(C)C CCC(CC)(CCC(=O)N(C)CCNC(C1CNC(=O)C1)=O)[N+](=O)[O-] C(C(F)(F)C(=O)N1CCCC(n2cc(CO)nn2)C1)NCC(=C1CCCCCC1)C C=CCCCC(C(=O)NCc1cc(C)cc(F)c1)NC(=O)COCC=C CCC1=C(C(=O)N2CCCC(NC(C3(C(C)C)CNC(=O)C3)=O)C2)SCCO1 C1(CNC(CC(=C)C)=O)CCC(F)(CNC(C2COCCN2C2CCCC2)=O)C1 N1(C(CC(CCC(CC)C)O)=O)CCCC(C2CCN(C(c3cscn3)=O)C2)C1 c1(C(=O)OC)cc(F)c(C(N2CC=CC(NC(C3CCCS3)=O)C2)=O)cc1F C(C(C)(O)C(F)F)NC(CN(C(=O)CC1CC=CC1)CCOC)=O C(=O)(C1=C(Cl)CCOC1)N1CC(C)CC(C(=O)NC(C2(O)CCC2)C)C1 N1(C(=O)C(O)CNC(C23CC2CNC3=O)=O)CCOC2C(O)CC12 c1(C(N(CCOCCNC(C=CSC)=O)C)=O)ccc(-n2ccc(C)n2)cc1.C(C)(=O)O C(C)(CCCCNC(=O)COc1ccsc1)NC(C(C)OCCC#C)=O C1(N)CC2(C1)CC21CCC1.C1(CNC(=O)NCCn2ccnn2)(C)CC12CCC2 CCCC(CNC(=O)C(F)CCC(=O)OC)C(=O)NC(C)CC.C(CC(=O)N)N NS(=O)(=O)c1c[nH]c(C(=O)NC2CC3CC2N(C(c2ccccc2CO)=O)C3)c1 C(C(=O)NCC(O)CNC(=O)CCc1cc(C2CC2)nn1C)(C(C)(C)C)OC N1(C(c2cnc(CCCC)s2)=O)CC2(C1)CN(C(C1CCSC1)=O)C2 N1(C(Cn2cnc(C)c2C)=O)CCCC2(NC(=O)NCc3ccccc3)CC2C1 N1(C(C(N)=O)=O)CCC(C(=O)NC2CC2c2ccccn2)C(F)C1 C1(=CC(=O)N(C2CN(C(CNC)=O)CC2O)C)CN2CCC1CC2.C(=O)(CS)OC N1(C(C2(OC(C)=O)CC2)=O)CCC(C)(C)C(CNC(=O)CC2(C#N)CC2)C1 CC(C)CC(F)C(=O)N1CCC(CN(C)C(c2cnn(CCO)c2N)=O)C1 C1(NC(c2c(CC)cccn2)=O)(CC)CCCN(C(c2ccnc(C)c2C)=O)C1 N1(c2ccsn2)CC(C)(C)OC2(CCOC2)C1.CC(O)CC(C)c1ncno1 C1(C(N2C(C3(O)CN(C(CN(C)C)=O)C3)CCC2)C2CC2)CCC(F)CC1 CC(C)CC(C(N)=O)NC(=O)C(C(C)(C)C)NC(=O)CCc1cnoc1 N1(C(CC(CC)C2CCC2)=O)CCOC(CCNC(=O)CCC2CCCO2)C1 N1(C(CCc2cnc(C)o2)=O)CCN2CCN(C(=O)CNC(=O)C3CC3)CC2C1 c1(CC(N2CCN(CC(=O)NCCC(C)(C)O)C(=O)C2)=O)ccc2[nH]ccc2n1 C1(C(=O)NC2CN(C(c3ncc(Cl)s3)=O)C2)CCCCCC1(F)F Cc1cnncc1C(N1CCC(C2CCCN2C(=O)CCc2ccco2)C1)=O C1(C)(C(=O)NCC(CC=C)NC(=O)C=CC=CCC)CCCC1(F)F CC(O)C(C(=O)NCCNC(N)=O)NC(c1occc1CO)=O S(=O)(=O)(c1cnc(NCCCc2ccccc2)c(Cl)c1)NC(CC)COC CCC(CC)CCCC(=O)N1CC(NC(C2CSCN2CC2CCC2)=O)CC1C C(=O)(C1=NOC(C)(C)C1)N(C1CCN(C(C2CN(CC)C(=O)N2)=O)CC1)CCO Cc1nc(NCc2coc(C)n2)cc(=NCc2cccn2C(C)C)[nH]1 c1(C(N2CCC(CCNC(c3ccoc3)=O)CC2)=O)cc(Br)cnc1Br c1(CC)nc(N2CCC(NC(=O)C(O)C(C)(C)C)C(O)C2)cc(C)n1 C1(O)(CCNC(=O)C2CC2)CCN(C(C2C(c3ccccc3)C2(F)F)=O)C1 C1(CNC(C2(C)CC(C)C2)=O)CCN(C(=O)CCCn2ccnc2)C(C)C1 c1(CC(=O)OCC)ccc(C(=O)NCC2CCC(C)O2)cc1.c12cn(nn1)C2 c1(NC(=O)NCC2N(CC)C(=O)CC2)cc(C)c(F)cc1I CCC(C)CCC(=O)NC1CC(OCC(=O)Nc2ncccc2C(C)C)C1 c1(OC)cc(C(=O)N(C)CC2CCN(C(C3CCCC(F)C3)=O)CC2)ccc1F c1(C(=O)NCC2CC(NC(c3ncn(C)c3)=O)C2)cc2n(c1)CCC2 C(=O)(C1=NNC(=O)CC1)N1CC(N(C)C(C2CC2[N+](=O)[O-])=O)C(O)C1 N1(C(C2(O)CCCC(C)(C)CC2)=O)Cc2nccn2CC(OCc2ccccc2)C1 C1(NC(=O)Cc2nncs2)CC2CC(NC(c3ocnc3C3CC3)=O)C1C2 CC1CC(C)N(C(c2cccc3nsnc23)=O)CCN1C(c1ccccc1Cl)=O c1(CN2CCC(OC)C2)ncc(C)c(O)n1.C12(NC(C3CC3)CC)CCCN(CC1)C2 N1(C(c2ncn(C)c2)=O)CCN(C(c2scnc2C(F)(F)F)=O)CC1 C(C(C)(C(=O)NCCCC1CN(C(=O)CO)CCO1)OC)OC Cc1cccc(CN2CC3CCC2C3C(=O)NCc2ncc(C(=O)O)cn2)c1F N1(C(C=C(CNC(c2c(OC)nsc2)=O)C)=O)CCC2(CC1)N=N2 C(c1cn(C)cn1)=CC(=O)N(C(C)C(=O)N(C(C)C(C)C)CC)CCC S(=O)(=O)(c1ccccc1Cl)N1CC2C(CNC(c3cc(Br)ccc3F)=O)(C2)C1 c1(C(N2CCC(NC(c3nc(Cl)c(Cl)s3)=O)(CO)C2)=O)ccn2nccc2c1 C(CCCCn1cc(C2CC2)nn1)C(N1CCC(Sc2ccccc2)C1)=O C(=O)(C1=CCC(C)CC1)N(CC(CN(C(CCc1ccnc(C)n1)=O)C)O)C c1(SC)ncc(C(=O)NC2(CO)CN(C(=O)C(C)Cc3ccccc3)C2)s1 C1(NC(C(CC)OCC)=O)CN(C(=O)CN2CC3CC3C2)CC12CC2 N1(C(C2CCC(C)(CC)O2)=O)CC2CCC2(N(C)C(c2ccc(OC)cc2)=O)C1 N1(C(c2c(SC)ccs2)=O)CCCC(C)C1CCNC(=O)C1=NNC(=O)C1 c1(C(=O)NC2CC(F)(CNC(CN3CCC(C)C3)=O)C2)ccccc1OCF c1(C(=O)NC(C)CNC(c2cccc3c2COC3)=O)ccc2nc(O)cn2c1 N1(C(C2CCC3N(C(CCC=C(C)C)=O)C2CC3)=O)CCOc2ccccc21 c1(C(=O)NCC(CC=C)NC(C2CS(=O)(=O)C2)=O)c(C)ccc2nsnc12 c12coc3c1CN(C3)C2=O.c1(NC(CC=CC(C)(C)C)=O)cc(C2CC2)on1 C1(OC)CC2CN(C(C3(C(C)C)CCCN3C(=O)C(F)C3CCCC3)=O)CC12 c1(CC)ccc2cc(C(=O)NCCC3CSCCN3C(=O)COCC)ccc2c1 c1(C(N2C(C(=O)NC(c3ccn(C)n3)CC)CC2)=O)nccc2cc[nH]c12 n1(CC(=O)N(C2CCCN(C(=O)C(=O)N)C2)C2CC2)ncc(C)cc1=O.CO c1(NC(N2CCN(CC)CC2)=O)c(OC)ccc2ncccc12 c1(C(=O)NCC2(O)CC(CNC(=O)CCCC3CC3)C2)cc2ncccc2[nH]1 C1(NC(c2ocnc2C2CC2)=O)CC12CCN(C(=O)CS(=O)(=O)C1CC1)CC2 N1(C(c2c(C)nc(NC(C)=O)s2)=O)CCOCC(NC(=O)C2=NOCC2)C1 C(=O)(C(C1=NOC2CC12)N1CCN(c2ccc(C)cc2)C(=O)C1)NC(CC)(C)C c1(N(C)Cc2c(Br)cn(CC)n2)ccc(S(=O)(=O)NC2(CC)CCOC2)cc1Br c1(C(c2nnnn2CCCF)NC2(C=C)CCC2)cccc(OC)c1Cl N1(C(c2c(CC)n(C)nc2)=O)C2CCC1CC(N(C)C(c1cnnn1CC)=O)C2 C#CCC(C(=O)NC1CCCC(O)C1)NC(=O)CNC(=O)CN(C)C c1(CC(=O)NC23CC2CN(C(=O)CN2C(=O)CCC2=O)C3)cc(F)ccc1F c1(OC(C)=O)ccc2[nH]cc(C(=O)Nc3ccc(C4NC(=O)NC4=O)cc3)c2c1 C1(C(=O)NC2(CNC(C3CC(N(C)CC)C3)=O)CC2)CCN(C)C1C N1(C(CNC(N)=O)=O)CCC2(NC(c3ccc(F)c(C(F)F)c3)=O)CCCCC12 C(CCC(=O)NCc1csc(CNC(C23CCC(C2)C3)=O)n1)NC=O Cc1ccc(CC(=O)N(CC(O)CNC(=O)CCCc2ccc(C)s2)C)cc1O N1(C(c2cc(C)ns2)=O)CCC2CCC12CNC(=O)C#CC(C)C C1(NC(=O)CC2CC2)CN(C(c2cnc(S)n2-c2ccccc2)=O)C2(CCC2)C1 C(CO)(CC(F)(F)F)NC(CCC)C(c1nnnn1-c1cccc(OC)c1)OC c1(CCC(=O)N(C2CCN(C(C(CC=C)C)=O)C2)C)ccc(Cl)c(OC)c1 Cc1cc(C(N2CCCC(C(C)C(=O)NCC3(O)CC(C)(C)C3)C2)=O)cnn1 c1(NC)nc(C)ccc1C(N1CCCCC1CN(C(=O)Cc1nnc(O)s1)C)=O Cc1cc(C(=O)NCC2(NC(c3ccns3)=O)CCOCC2)[nH]c1C c1(CC(C)C(=O)NC2CC2CNC(C2CCO2)=O)ccc([N+](=O)[O-])cc1 c1(C(N2CCC(CN(C(CCOC(C)=O)=O)C)C2)=O)ccc2c(c1)CCCO2 c1(SC)ccc(O)c(C(N2CC3C(CNC(=O)CCc4cccnc4)C3C2)=O)c1 N1(CC(=C)Br)CCC(N2CCN(C(=O)CCc3ccc(OC)cc3)CC2)CC1 c1(C(=O)NC(CC)C(F)(F)F)cnc2n1CCN(C(C1(C)COC1)=O)C2 N1(C(C2(C)CC(F)(F)C2)=O)CC(NC(=O)C2=COCCO2)CC(F)C1 C1(C2CN(C(=O)C(O)Cc3ccc(Cl)cc3)C2)(NC(c2[nH]ccc(=N)n2)=O)CC1 c1(NC(COC2CCN(C(CCc3cccc(C)c3)=O)C2)=O)cc(Cl)c(O)nn1 N1(C(CCc2c(C)n[nH]c2C)=O)CC2CC(NC(=O)Cc3nc[nH]n3)CC(C2)C1 C1(O)(C(C)(C)C)CCN(C(=O)C(=O)NCCCCC#N)CC1.C1(=O)CO1 C1(COC)(CNC(=O)Cc2ccccc2Cl)CCCN1C(C1CC1(Cl)Cl)=O CC1CCN(C(c2cc(=O)cc[nH]2)=O)C(CNC(c2ccccc2)=O)C1 CC1CC(CC(=O)N(C)CC2CCCN2c2cc(Cl)ncn2)CC(C)(C)C1 C1(NC(c2cccc3ncnn23)=O)CC(C2CCN(C(C3(SC)CCC3)=O)C2)C1 Cc1cc(N)c(C)nc1C(=O)NC1CCN(C(c2cc3nccnc3[nH]2)=O)C1 CC(C)(CC(=O)N1CCOCC1C(F)(F)CO)C1CC1 O=C(C1=NOC2COCC12)NCC(N1CCCc2occc2C1)=O C(C1CCOCC1)=CC(=O)NC(C1CCOC1)CNC(CC=C(C)C)=O C1(NC(C2C(CC)C2)=O)CCN(C2CCN(C(=O)CCC(C)OC)CC2)CC1 C1(NC(C2(CCC)CCC2)=O)CC1C1CCN(C(c2ccnn2C(F)F)=O)CC1 N1(C(CC2(C)CCOC2)=O)CCC2(CCN(C(c3occ4c3CCC4)=O)C2)C1 c1(C(=O)NCC(O)C2CCC2)ccc(F)cc1.C1(C2CCCO2)C(=O)N1C1CCC1 c1(OCC(N2CCC3CN(CCOc4ccccc4)C23)=O)cccc([N+](=O)[O-])c1 C1(C(=O)NCCC(C)N(C(C(C)(C)OC)=O)C)CC12CCc1ccccc12 c1(OC)ccncc1C(=O)NC1CCC(NC(c2cnccc2C(F)(F)F)=O)C1 C(C(C)(C(C)C)NC(c1cn(-c2ccc(F)cc2)nc1C)=O)NC(CC=CC)=O N1(C(c2cc(COC)on2)=O)CC(NC(=O)CC2(C)CCCO2)C2CCCC12 N1(c2nccc(OC)n2)CC2CCCC(NC(CCOCC#C)=O)C2C1 C1(NC(=O)C=Cc2cncnc2O)CC(O)CN(C(=O)CN2CCCCC2)C1 c1(C(=O)NCC2(CNC(C3(O)CCC(CC)C3)=O)CCC2)cc(N)cnc1Cl C1(NC(c2cccc(N)c2)=O)CN(C(=O)COc2ccsc2Cl)C2(CCOC2)C1 C1(CN(C(CCNC(=O)NC)=O)C)CCCC1NC(=O)CC(Cl)Cl CC1CCn2cc(C(N3CCOC(CNC(=O)CN4CCOCC4)C3)=O)nc2C1 Cn1cc(Cl)cc1C(=O)NC1CCCN(C(C2(C(F)F)CCCCC2)=O)C1 C1(NC(C(C=CC)O)=O)CC(CNC(=O)CC(F)F)CC1O N1(C(CC=CCC)=O)CCC(C)(C)C(C(=O)NC(C)CC(C)(C)OC)C1 Cc1noc(C)c1C(C)C(=O)NCC1CC(C(=O)N(CC(O)CO)CCO)CO1 c1(-n2ccc(C)n2)ccccc1CN1CC2C(CNC(C3CCSC3)=O)C2C1 N1(C(CCCCSC)=O)C2CCC(C(N3CCC(c4cnco4)C3)=O)C1CC2 CC1C(NC(c2ccc(O)nn2)=O)CCN1C(=O)Cc1cnccn1 N1(C(Cn2cnc(=N)[nH]2)=O)CC(=O)CC1C(=O)NC(CO)C1CC1 CC(C)CC(F)C(=O)N(C)CC1COCCN1C(c1ccc(F)cc1Cl)=O N1(C(c2ccc(C(F)(F)F)c(O)c2)=O)CC2CC1CN(C(C13CC(F)C1C3)=O)C2 c1(C(=O)NC2C(C(=O)Nc3nc(C)nc(Cl)c3)CCC2)ccc2cncn2c1 C(=O)(C(CN)C(C)(C)C)NCC(c1ncc(F)cn1)(C)C C1(CC)C(NC(=O)CN(C)Cc2ccccc2)CCN1C(c1cc(C#N)c[nH]1)=O C1(C(=O)NCC(C)NC(=O)C(C)(C)C)C[Si]2(CCCC2)CN1C(N)=O c1(C(=O)NCCC(C)N(C)C(c2cncc(F)c2)=O)cc(S(C)(=O)=O)co1 N1(C(c2c(Cl)cn(CCC)n2)=O)CCC(C)C(N(C)C(c2ncncc2C)=O)C1 c1(CC)c(C(=O)NC2CCCC2(C)NC(=O)Cn2nccn2)sc2ccccc12 C(=O)(CCC(=O)NCCC)NCC1C(C(=O)NCC(=C)Cl)CCC1 C1(C(N2CCC(C(C)(C)NC(C3CC34CCC4)=O)CC2)=O)CN2CCN1CC2 CC(C)(C)C1CCNc2c(C(=O)NCCCP(C)(C)=O)cnn21 C1(C(=O)NCc2c(C)c[nH]n2)CCN(C(=O)C(C)C2CC2)C12CC2 CCCCC#CC(C)(C)NC(c1cc(CNC(c2ccc(C)c(F)c2)=O)nn1C)=O c1(CC)cccc(C)c1C(=O)NC1CC(CCNC(=O)C(=O)NC(C)=O)C1 C1(C(=O)NC(CNC(Cc2nc(C)oc2)=O)(C)CC(C)C)CCc2nnnn2C1 c1(C(=O)NCC2C(NC(C(C(C)(C)C)SC)=O)C2)cc2n(c1)CCCC2 O=C(CC1OCc2ncccc21)NCC1CCC(CNC(C2(O)CC2)=O)CC1 N1(C(C(CCCCC)O)=O)CCCC(C2CCCN(C(=O)CCC[N+](=O)[O-])C2)C1 C(=O)(C(F)(CC)C(=O)OC)NCC1(NC(C2(CC)CC2)=O)CC2CCC1C2 c1(C(=O)OC)cc(C#N)ccc1NC(C1CCN(Cc2cc(Br)c[nH]2)CC1)=O C12(NC(c3ccnnc3O)=O)CCCC1N(C(=O)CCOCC1CC1)CCC2 C(C(O)C(=O)N(CC(C)C(=O)N1CCC1CN=[N+]=[N-])C)SC C1(CNC(CCCC#N)=O)C2CCC(C2)N1C(=O)CCOCc1ccccc1 C1(COC)CC2(CCN2C(=O)CNC(c2ccc(C(C)=O)o2)=O)C1 N(C1CCCn2nncc21)C(C(=O)NCC(c1ccccc1F)C)=O C1(C(=O)NCC=CC)CCCCN(C(c2c[nH]c(C)c2)=O)C1 c1(C(=O)NCc2ccnc(OC3CCCC3)c2)cc2ccc(O)nc2s1 C1(NC(C(C(CC)CC)C)=O)CN(C(C2CCCC3CC23)=O)C2CCCCC12 c1(C(N2CC(C(C)NC(CC(CC)O)=O)C2)=O)cc([N+](=O)[O-])ccc1OC c1(C(=O)Oc2ccccc2)cnc(CN(CC(C)CC2CCC(F)C2)C)cn1 Cc1c(Br)ccc(O)c1C(=O)N(C(C)CNC(=O)C(O)Cn1cncn1)C C1(NC(C=CC(C)C)=O)CCC(NC(=O)CC(C)N(C)C)CC1 C(=O)(C(CCOCCO)NC(C1CCCNC1=O)=O)N(CCN(C(C)=O)C)C CC(N(C)N1CCc2c(Cl)ccc(Br)c2C1)c1nccs1 C(=O)(C(CC(F)F)C1CCC1)N(C(CNC(=O)CC(C)(O)C=CCl)C1CC1)C c1(OC)ccc(C(F)(F)F)cc1CN1CCC(C)(C(=O)Nc2cncnc2Cl)C1 c1(C(=O)NCC2CCC(C)N(C(c3ncc(F)cn3)=O)C2)cc2ccccc2s1 n1(CC)nc(C(c2nnnn2CCOC)NC2CC(F)(F)C2)c(Br)n1 C1(NC(C(CC)OCC)=O)CCN(C(c2csc(=N)[nH]2)=O)CC(C)(C)C1 N1(C(COC)=O)CCC(O)C(C(N2CC3CCC2CO3)=O)C1 Cc1ncnc(O)c1CCC(N1CCC(Nc2ccc(C(C)(C)C)cn2)C1)=O N1(C(c2c(CC)n[nH]c2)=O)CCCC(NC(=O)C=Cc2nc(C)c(C)[nH]2)CCC1 N1(CC(N2CCCC(N(C(=O)CSCC(N)=O)C)C2)=O)CCc2ccccc21 c1(OC)cc2c(cc1OC)C1(CC1)CN(C(C1CCC(C#N)(OC)CC1)=O)C2 Cc1ncnc2c1CC(C(=O)NCC(C)(C(C)C)NC(=O)COC(C)(C)C)CC2 N1(C(c2cccc(OC)c2F)=O)CC2CCN(C(=O)C=CC(F)(F)F)C(C2)C1 C1(NC(C2(C)CC=CC2)=O)CC2(CCCN(C(=O)CCn3cccc3)C2)C1 c1(COC(C)C)ccc(C(N2CC(NC(=O)COC3CC3)CC2C)=O)cc1 C1(CC)(CC)CC(NC(=O)CC(CN(C)C)CC)CN1C(=O)C1=CCCCO1 CCCC(C(=O)N1CC(O)(C(F)C(=O)NCc2ccc(=O)n(C)c2)C1)C(C)C C(=O)(CCS(=O)(=O)Cc1ccncc1)NCCC(C)NC(=O)C(=O)NC1CC1 C1(CNC(C(=O)NCCOC)=O)CC2(CCN(C(=O)CCC(C)(F)F)C2)CO1 C1(NC(c2csc(-c3ccccn3)n2)=O)CCN(C(C2(F)CC=CC2)=O)CC1F N1(CCNC(C(C2CC2)NC(c2c(OC)ccs2)=O)=O)CCCOC1=O C1(CCN(C)C(C2(C3CCC3)CC2)=O)CCCCN1C(C1C2CCCCC12)=O c1(C(N2CC(C(N(C)CC3CC(F)C3)=O)C2)=O)cc2ccccc2n1C Cc1cc(C)n2nc(CC(=O)N(C)CCNC(c3nocc3C)=O)nc2n1 Cc1ccnnc1C(N1CC=CC1CNC(C1CC(C)(C)CO1)=O)=O c1(N(c2nnc(COCC)n2CCOC)C)cc(Cl)ccc1C CC(C)(C)C(O)C(=O)NCc1cn(C2CCN(C(=O)CCF)CC2)nn1 N1(C(CNC(C(CC)C)=O)=O)CC2CCN(C(C3CC(C)(O)C3)=O)CC12 c1(C(=O)NCC2COCO2)csc2c1CCN(C(c1cnnc(Cl)c1)=O)C2 c1(C(=O)NC2C(NC(=O)Cc3cnsc3)CCC2)ccc(Cl)cc1O c1(CC(=O)N(C)CCC2CCN(C(C3CC3F)=O)CC2)csc2cccc(F)c12 C(C(C)C(=O)NCc1ccoc1C(=O)NCC(C1CCC1)O)OCC Cc1cnc(Br)c(NC(C2CCC(NCc3c(Cl)cncc3Cl)C2)=O)c1 C1(NC(CCC=CC)=O)CCN(C(=O)CC2CC2c2ccccc2C)C1C1CC1 C1(C(N2CCC(F)(C(=O)NC3CC(C4CCC4)C3)CC2)=O)CCCC12CCC2 C1(CCOC)CN(C(C2(C=C)CC2)=O)CCN1C(C1CC(F)(F)C1)=O c1(NC(C(c2cccc(C)c2)NC)=O)ccc(C2CCCCC2)cc1F C1(C(N2CC(NC(C=Cc3c(C)ncs3)=O)C(C)C2)=O)CC2(C1)CC(O)C2 C12(CC(=O)NC3C(NC(c4cnc(C(C)OC)s4)=O)C3)CCC(CC1)OC2 O=CCNCC=CBr.C(=O)(CSC)NC1CCC1 c1(OC)ccc2c(c1)NC(=O)C2CCNCC(O)COc1ccc(F)c(Cl)c1 c1(OC)ccc(Cl)c(C2CCCN2C(=O)NCCC(C)(C)C)c1 N1(C(C2(NC(=O)CNS(N)(=O)=O)CCN(C)C2)=O)CCC(C2CCCC2)C1 c1(OCC#N)cccc(C(=O)NC(CC(=O)O)C2CC2)c1 c1(CC(=O)Nc2ccno2)ccc2c(c1)CN(Cc1c(F)cccc1I)CC2 N1(C(c2cnc(CC)s2)=O)CC2CC(C1)C2NC(=O)C(C(C)CC)NC(C)=O C12(CNC(c3cccc(-c4ccc[nH]4)c3)=O)CC1CN(C(=O)CC1C=CCC1)C2 c1(CCCC)nc(COC)c(Cl)[nH]1.C1(CN)CCCCN1C(=O)CC1CCC1 C=CCC(CNC(=O)CC1CCCN1C)NC(=O)CCc1cnc(C)s1 C(CC(F)F)(C(=O)NOCCc1ccccc1)NC(c1c(C)cc(F)cc1)=O C(=O)(C(CCC1CC1)NC(=O)C(N1CCCCC1)C)NCC1ON=C(C)C1 C1(NC(C2(CCCC)CC2)=O)CC2CC(C1)N(C(c1c(Cl)n[nH]c1C)=O)C2 c1(C(=O)NC2(CNC(C3C(C)CC3)=O)CCOCC2)cc(F)c(CO)c(F)c1 C(C(=O)NCC1CC1NC(=O)C(c1cncc(F)c1)C)(C(C)C)OCC(C)C N1(C(CCC#CC)=O)CCC2(CC1)COC(CNC(=O)C(C)CN(C)C)C2 C12(CNC(=O)CCC3CC3)CCCN(C(c3ccc(SC(F)F)cc3)=O)C1C2 N1(C(CCCOCCC)=O)CCOCC2(CCOCC2)C1 C1(NC(C(CC#C)C2CC2)=O)CN(C(c2cccc3cncn23)=O)CC2(CC2)C1 Cc1cccc(C)c1CNC(=O)C(c1cnc(Cl)s1)N(C)C(c1ccco1)C CN1CCN(C(=O)CC2CCOCC2(C)C)C(CNC(=O)C(F)=CCCF)C1 C1(NC(c2cscc2Cl)=O)CN(C(c2cc(F)n[nH]2)=O)C2(CCCCC2)C1 c1(C2(C)CCO2)cccc(CN(Cc2cccs2)CC2CCCO2)c1 CN1Cc2ccccc2CC1C(=O)NC1CC(CO)C(O)C(O)C1O.C12CCN1C2 C1(NC(=O)C(c2cc(F)cc(F)c2)O)CCC2(CCN(C(=O)C(F)(F)CO)C2)C1 C1(NC(CCC=C)=O)CC1C1CCCN(C(C2(CF)CC3(CCC3)C2)=O)C1 C1(C(N2CC3(CC(NC(C4CC5CC5C4)=O)C3)C2)=O)CCCCC12OCCO2 C1(CNC(=O)CN2CCCC2CO)CN(C(=O)COC(F)(F)F)CC2(CCC2)O1 C(C(=O)N1CC(N(C)C(=O)C2CC2)C(CO)C1)(C(C)(C)C)NC(C)=O C1(CNC(C2C(CC)C2)=O)CN(C(C23CCCC2C3Br)=O)CCC1(C)C C1(CNC(=O)Cc2cn[nH]c2)CC(NC(C2(Cl)CC2(F)F)=O)CC1O O=C(C1CC=Cc2ccccc21)NC1CN(C(=O)CCF)CCC1F N1(C(c2cccc(Cl)c2)C(=O)NCCCOC)CCOC(C)(C2CC2)C1 C1(C=O)CCn2nnnc2C1.n1(CC2CC(=O)C2)cc(C(=O)NC2(C)CC2)nn1 C1(C(=O)NCC(CC)(C)O)(NC(=O)CCc2cncn2C)CCCCC1 C1(n2cc(-c3cn(CCC)nc3)nn2)CC2CCC1(NC(c1cnc(C)s1)=O)C2 C1(CNC2CC(C(c3[nH]cc(C)c3)NC(=O)CCCC3CC3)C2)CC2CCC1CC2 Cc1ncc(CC(=O)NC2CCN(C(c3c[nH]c(=N)nc3O)=O)CC2C)c(O)n1 C(C)(CS(C)(=O)=O)N(CCC1CCOCC1)Cc1n(CC)ccc1 c1(C(=O)NC2C(NC(CCCN(C(C)C)C)=O)C2)cc(Cl)cc(C(F)(F)F)n1 C(CC(CC)C(=O)N(C1(CC(N2CC(O)(CC)C2)=O)CC1)C)=CC CCCCS(=O)(=O)CC(=O)N1CC=CC1CNC(C1CCC2CC1C2(C)C)=O N1(C(C(CC)(C)C)=O)CCC(C2CCN(C(c3cncn3C)=O)CC2)C1 N1(C(C(C(C)C)(C)C)=O)CCN(C(=O)C(OC(F)(F)F)=O)CC(C)(F)C1.CO N1(C(C(CC)NC(=O)C(=Cc2ccccc2)C)=O)CC(=O)N2CCCC2C1 C1(CC)CCCCCCN1C(C1C(C)CN1C(C1CC2CC1CC2=O)=O)=O c1(C(=O)NCCCC(C)NC(=O)C(C)(C)C(N)=O)ccc([N+](=O)[O-])s1 c1(C(=O)NC(C2CCN(C(=O)C(F)C3CCC3)CC2)C)cn(C)nc1Br c1(C(N(C)CC2(O)CCCN(C(COC(C)C)=O)C2)=O)cc2ccnn2cn1 C1(C(=O)NC2COC(=O)C2)(COC)CCCN1C(=O)Cc1ccccc1 c1(C(N(CCNC(=O)Cc2cccc(OC(F)F)c2)CC)=O)cccc(F)c1O CC(CN(C)C)CC(=O)NCC(C1CCN(C(=O)CC2CCCN2C)CC1)(C)C c1(C(=O)NC2C(NC(=O)CCOCC(F)(F)F)CC2)cccc2c1COC2 O=C(C#CC1(C(=O)O)CC1)NCC=CCNC(c1cnns1)=O C1(C(N2CCC(CC=C)C2)=O)CN(C(c2ccsc2OC)=O)CC1F C1(C)(NC(C(C=CC)O)=O)CCCN(c2ccncn2)C1 c1(OC)cccc(-c2nc(-c3c[nH]c(C#N)c3)n(C34CCC(OC)C3C4)n2)n1 Cc1ccnc(COC(c2ccsc2C)=O)n1 C1(C(=O)NC2CC(NC(=O)CCCN3C(=O)CNC3=O)C2)CC2CC(=O)C1O2 C1(NC(CN(C(C)=O)C)=O)CCC(NC(=O)C(F)(F)c2cccnc2)C1 NS(=O)(=O)c1csc(C(=O)NC2C3CC(NC(c4csc5nccn45)=O)CC23)c1 c1(CNC(N(C(C)CO)C2CC2)=O)[nH]c(=N)nc(O)c1Br C(C)(C(=O)N1CCCC(C)(C(=O)NOCCC(C)O)C1)(C(C)C)OC CC1CN(C(=O)CCN2CCC(F)C2)CC1NC(=O)CC1(O)CCCC1 CN1CC(=O)Nc2cc(C(N3CCCN(C(c4ccoc4)=O)CCC3)=O)ccc21 C1(C)CCC2(CC1)COC2.c1(NNC(=O)CSCc2cnc[nH]2)ccc(F)cc1 CC12CCCOC1CN(C(=O)Nc1cc(OC(F)(F)F)ccc1F)C2 C1(CC(=O)NCC(CN(C)C)O)C2CCC(C2)N1C(=O)CC1CCCN1C c1(OC)ccc(CNC(C2CC2C(=O)NC2CCN(C3CC3)CC2)=O)cc1O Cn1c(C(=O)NCCOCCNC(C2(Cl)CC2)=O)cccc1=O N1(C(CCC(c2ccc(C)cc2)=O)=O)CC2CC3CC2C1C3NC(C1CC1C)=O N1(C(c2ccc(Cl)cc2)=O)CCCC(C2CN(C(c3conc3C3CC3)=O)C2)C1 C(=O)(C#CC1(C)CCCO1)NC(C1CCN(C(=O)Cn2nnc(=N)[nH]2)CC1)C C(N(C1CC1)N1CCC(C(=O)N)CC1)C1OCC(C)(C)OC1.c1ccccc1F Cc1cc(C)c2nc(N3CCC(C)C(NC(c4cnc(C)s4)=O)C3C)sc2c1 Cc1nccc(C(N2CC3CC(NC(=O)CCSc4nnnn4C)C2C3)=O)c1C c1(C(N2C(C(C)NC(C(CC)N(CC)CC)=O)CCC2)=O)cc(C(C)C)n(C)n1 c1(C(=O)NCCCCCN(C)C(C2(C)CCCC2O)=O)ccc([N+](=O)[O-])s1 C1(CC)(NC(C2CCC3(CC2)CC3)=O)CCCN(C(c2cn(C)nc2OC)=O)C1 c1(C(=O)OC)c[nH]nc1C(=O)NCC1CC(NC(=O)CCC2CCOC2)C1 c1(C(N2CCC(CNC(c3c(OCC)n[nH]c3)=O)C2)=O)cccc2nc(C)[nH]c12 C1(NC(c2c(C)cno2)=O)CN(C(C2CN(C)CCO2)=O)C2(CCC2)C1 C1(OC)(CNC(=O)Cn2ccnc2C(C)C)CCN(C(C2CCSC2)=O)CC1 N1(C(c2cccc(C#C)c2)C(=O)NCC2CC2)CCOc2ccc(Cl)cc2C1 C1(C)(C(=O)NCC23CC(NC(C(c4cnccn4)C)=O)(C2)C3)CC(C)(C)C1 c1(C(=O)NC2CC(C(C)NC(C3CC3CF)=O)C2)ncncc1Cl C1(C(N(C(CN(C(c2cccc(COC)c2)=O)C)C)C)=O)Cc2nccn2C1 CCCC(C(N)=O)NC(C1CCC(C(C)C)N1C(=O)CC1CCCC(=O)C1)=O C1(C(N2C(CCC(=O)Nc3cc(Cl)no3)CCC2)=O)C2CCC(C2)C1CO Cc1ccc(Cl)c(C(N2CCCC(CCNC(C3CCNC3)=O)C2)=O)c1 c1(COC)ccccc1C(=O)NC(C1CCCN1C(=O)C(C)(F)F)C N1(C(c2n(C(C)C)ncc2Cl)=O)CCC(C)C(CNC(=O)CCc2nncs2)C1 C1(CNC(C(=O)NCC(C)(C)OC(C)C)=O)CN2CCC1(F)CC2 N#Cc1ccc(N)c(C(N2CCC(CNC(C3(C4CCC4)CC3)=O)C2)=O)c1 S(=O)(=O)(c1ccc(Br)cc1N1CC(O)C(C2CC2)C1)N(C(CCSC)C)C C(=O)(C(O)CC(F)(F)F)NCC1(CO)CCN(C(C2N(CC)CCOC2)=O)CC1 c1(C(=O)NCC2N(C(C3C(OCC)C3)=O)CCCCC2)cc2scc(C)c2[nH]1 c1(SC)nc(N2CCCC(NC(c3ccc(CO)o3)=O)C2)cc(C)n1 N1(C(CC(n2c(CC)ncc2)C)=O)CCC(=O)N2CCCC12 CC1(C)CCCOC1C(=O)NC1CC(O)C1CC(=O)NCCc1cncnc1 c1(C(=O)NCC2CCCN(C(C(CCC=C)(F)F)=O)C2)c[nH]c2ccc(O)cc12 c1(CC2CCC(C(=O)O)CC2)cc(CN2CCC(O)(C(=O)O)C2)ccc1F C1(C(N2CC(CCCCC)C2)=O)COCCN1C(c1cc(C)oc1C)=O c1(C(=O)NCC(C)(CO)NC(C(C)NC(C)=O)=O)ccn2nccc2n1 C1(C2CCCN(C(c3ccc(N)c(Cl)n3)=O)C2)(NC(C(C(C)C)C)=O)CC1 c1(CN2CCC(C(C)C(=O)NCC3CCCC(O)C3)CC2)ccc(F)cc1Cl C(=O)(C1=NOC(C)C1)N(CCC(=O)NC1CC(=O)NC1=O)CC=C C(=O)(C(C)S(N)(=O)=O)N1CC(C(C)C)C(C(N2CCCCC2C(C)(C)O)=O)C1 C1(NC(C(C2CN(C(CC(=O)N(C)C)=O)C2)O)=O)C2CC3C(C2=O)C13 c1(CC(=O)NCC2(F)CN(C(C(CC)c3cccnc3)=O)C2)cc(C)cc(F)c1 c1(NC(c2c(Cl)ncn2C)c2n(CC(=C)C)nnn2)ccc2sncc2c1 C(=O)(C(CC(F)F)N(C)C(C1CC1C(F)F)=O)NC(c1nn[nH]n1)CC N1(CCC(C(=O)NC(c2nsc(C(F)F)n2)C)F)C(=O)c2ccccc2C1=O c1(C(N(CCCNC(C2CCC(OC)C2)=O)C2CC2)=O)cc(Cl)c(F)cc1Cl c1(CC(N2CCC(NC(CCC3C(C)(C)C3)=O)C23CC3)=O)c(F)cccc1C#N CC1(C(N2CC(OCC(=O)NCCn3ncccc3=O)C2)=O)CCOCC1 N1(C(CCCOC)=O)CCCC2CCN(C(c3cnn4c3C(=O)NCC4)=O)CC12 N(C(=NCCCF)N1CCC(C)(COC)CC1)C(C#C)C(C)OC c1(CC)[nH]nc(C(=O)NCC2CCC(C(=O)NCc3cnccc3C)CC2)c1F C(=O)(C(CC(C)C)c1ccccc1)N1CC(N(C(c2cc(C)oc2)=O)C)C(O)C1 C1(NC(c2ncc[nH]c2=O)=O)C2CCC1N(C(=O)C(O)C1CCC1)C2 CCC1=NOC(C(=O)NC2CCCC2NC(=O)CN(C(=O)COC)C)C1 C1(NC(CN(c2cnccn2)C)=O)CN(C(=O)C2CC2)CC(F)(F)C1 C1(CCC)CN(C(c2nc(C)c(C)s2)=O)CCN1C(C1CC(CC)C1)=O CC(C(=O)N1CCC2(C1)CN(C(=O)CN1CC(F)(F)C1)C2)C(C)C(C)(C)C c1(C(N2C(C(=O)NCC3(C)CC(C)(C)C3)CSCC2)=O)ncc(F)cc1N c1(C(N2CC(C(N3CCC(OC)C3)=O)C2)=O)cc(CSC)c(C)s1 c1(C(=O)NC(CCC)C(=O)NC(CO)C(C#N)CC)c[nH]c2ncccc12 C(=O)(CC(C)(C)O)NCCC(CNC(C1C2(CC2)C12CC2)=O)OC c1(C(=O)NCC2CCC(F)(CNC(C(CCC)C)=O)C2)ccc(P(C)(C)=O)o1 C1(C(N2CC(CC(C)NC(c3cc(F)cnc3O)=O)C2)=O)CCCC(F)(F)C1 c1(NC(=O)CCS(=O)(=O)Cc2ccccn2)ccc2ncccc2c1Br C1(NC(C(CNC(C)=O)N)=O)(CO)CC(O)C(O)C(O)C1O CC1(C)CC(NC(c2ccsc2)=O)CN(C(C2(N(C)C)CCCOC2)=O)C1 c1(C(N2CC(NC(C3(Br)CC34CCC4)=O)C2)=O)cnc2ccoc2c1 c1(C(N2CCC(CCNC(C3CC(OCC)C3)=O)C2)=O)nccc2[nH]ccc12.COC N1(C(C2=CCN(C(C(C)C(F)F)=O)C2)=O)CC2(CCOC(=O)N2)C1 N1(C(C2(OC)CCSC2)=O)CCC2(CCCN2C(c2cc3cscc3s2)=O)C1 C(=O)(CCCC(C)(C)C)NCC12CC(NC(Cc3nc(C)[nH]n3)=O)(C1)C(C)O2 c1(C(N(CCCN(C(C(CC(C)C)(F)F)=O)C)C)=O)cccc2cc(O)ccc12 C=C(C)C(CC(=O)N1CCC(CC)(NC(=O)C(C)SCCCC)C1)OCC C#CCCCCC(=O)NCCC1CC(NC(=O)CSCC(=O)Nc2ccccc2)C1 C(=O)(C1CCc2cccc(F)c21)N1CCC(CNC(CCc2n(C)ccn2)=O)C1 N1(C(C(CC)N(C)C)=O)CCN(C(=O)CCNC(=O)CO)CC1C1CCC1OC c1(C(N2CCCCC(CNC(CCC(C)C)=O)CC2)=O)ccc(S(C)(=O)=O)nc1 c1(C(N2CC3C(CNC(CC(C)O)=O)(C3)C2)=O)csc2nnsc12 c1(N(CCCS(N)(=O)=O)C(C(=O)OC)Cc2ccccc2)cccc(OC(F)F)c1 N1(C(C(C=C)(F)F)=O)CCOC2(CCCN(C(c3cccnc3O)=O)C2)C1 c1(CNC2C(C(=O)NCc3cnccn3)C2)cc(Br)c(Cl)c(Br)c1 C(=O)(C(C)(C)C1CCN(C(=O)CC#N)C1)NC(c1nccn1C)C C1(CNC(C(CC)O)=O)CC2CCC1N2C(C1CCC(SCC)CC1)=O n1(CC=C)cc(CNC(=O)CCc2ccon2)nn1 c1(N(C)C)cc(Cl)ccc1Cn1cc(CN)nn1.C1(C)CCOC(=O)CC1 CCN(OC)C(=O)C(C)NC(C1CC2(CCC2=O)C1)=O C1(CNC(CC2C(C)C2(F)F)=O)(NC(C2CCC(C)(C)C2)=O)CCOCC1 c1(NC(C(C2CC=CC2)N(C(C)C(=O)N(C)C)CC)=O)ccc(Cl)cc1 Cc1cn2c(n1)CCC(C(N1CC=CC(NC(=O)Cn3ncccc3=O)C1)=O)C2 C1(C(C)C)CN(C(=O)C(C)SCc2ccc(Cl)s2)CCN1C(=O)C1=NOCC1 C1(CCOC)(CNC(C)=O)CCN(C(C2C=CCC2)=O)C1 c1(C(=O)NC(C(C)C)CNC(C2(C(=O)OC(C)(C)C)CCC2)=O)cc2n(n1)CCO2 C(C1CN(C(=O)CO)Cc2ccccc21)NC(C1CCC(CCCC)CC1)=O C1(NC(c2c(OC)c(Cl)ccc2)=O)CCC(O)CN(C(c2cnsn2)=O)C1 c1(C(=O)NC2CCN(C(CCNC(C)=O)=O)CC2)cc(N)c(F)cc1C c1(NC(C23CCC(CC2)N3)=O)cc(Cl)nc(C2CCCO2)n1 N1(C(C2C(C)N(C)CC2)=O)CCC(CNC(c2coc(Cl)c2)=O)C(F)(F)CC1 c1(C(N2CCCC(CC3CC3)C2)C(=O)NC2C(OC)CCC2)cc(OC)n(C)n1 C(CCC(=O)NCC1CC1(Cl)Cl)NC(CNC(=O)CCOC1CCCC1)=O C(C(C)S(C)(=O)=O)NC(C1(NC(C(C)CC2CCCC2)=O)CCSC1)=O c1(C(=O)NC2CC(NC(c3ccnnc3)=O)CC2O)n[nH]c2ccc(Cl)cc12 N1(C(c2c(NC)cnnc2)=O)CCOC2(CCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 C(c1nc(C)cs1)=CC(=O)NC1CC(N(C(CC)=O)C)C1 CC1CN(C(=O)C(=O)N2CCCC2)CCC1N(C(=O)C(O)CN1CCCC1)C C(CCCCC(=O)N(C)CC=CC(=O)NCc1cc(F)ccc1O)SC CCC(C)C(O)CNC(C1(CNC(=O)C(C2CCOCC2)=O)CC1)=O c12nnc3n1CCCC3C(=O)NC1CCCC1NC2=O.C1(CC)CCN(C)CC1 N1(C(C2C(=C)CC2)=O)CCC(O)C(NC(c2cccc(C(F)F)c2)=O)C1 C1(CNC(C2(NC(c3ncn4c3CCC4)=O)CCC2)=O)CC2CCCC2C1 N1(C(CC2(OC)CC2)=O)C2CCC1CN(C(=O)CNc1ccc(C(N)=O)cn1)C2 C1(NC(Cc2ccn(C(C)C)n2)=O)CC2(C1)CN(C(C1(C(F)F)CC1(F)F)=O)C2 Cc1cc(=O)n(C)nc1C(=O)NCC1(CNC(=O)C=Cc2ccsc2)CCCC1 CC1(C)OC2(CNC(C3CC34CCCC4)=O)CC1(NC(C1CCCCS1)=O)C2 C(=O)(C1CCc2cccc(O)c21)NCCCNC(COCCC(C)C)=O c1(C(C(=O)NC(CC)(C)CNC(c2cnc(CC(C)C)[nH]2)=O)=O)ccc(F)cc1 C(=O)(C(C)(C)Cn1cc(-c2cnccc2C)nn1)NC(c1ncccc1N)C N12CC3CCC(C1)N3Cc1ccc(Br)cc1C2=O.c1(CC)nccn1C C1(NC(C23CC(NC(CC4CC(OC)C4)=O)C(OC2)C3)=O)CC2CC1CC21CC1 N1(C(CCC(C)(C)C#N)=O)C2CC=C(C(=O)NCCCc3ccco3)C1CC2 CCC(C)CCCCC(=O)NCC(CO)NC(c1[nH]ccc1-c1ccccc1)=O C(N=c1nc(N2CCOCC2)[nH]c(=NC2CCCCC2C#N)[nH]1)c1cc(C)oc1 C(=O)(C1CCCc2ncnn21)N(C)CCC1CCCCN1C(=O)C(F)=C1CCC1 n1(CC)cc(C(=O)NCCC(O)C(=O)NCCOC(C)C(C)C)c(C)n1 CCC1(C)CN1.C(c1cnc[nH]1)=CC(=O)NC(C)C(=O)OC(C)C c1(NC(C(C)(C)CCNC(c2cc(F)ccc2O)=O)=O)ccc2c(c1)CCO2 N1(N(c2cc(Br)cn2C)C)CCc2[nH]nc(-c3nc(-c4ccccn4)nn3C)c2C1 N1(C(C(C)n2cccn2)=O)CCCC1(C)CNC(=O)Cc1cc(C(F)(F)F)no1 O=C1CCC(C(=O)NC2CCCCN(C(=O)CSc3cccs3)C2)n2cccc21 C(CCCCC(=O)NCC1(C(=O)NCC2NC(=O)CC2(C)C)CCCC1)OCC c1(C(=O)NCC2(O)CC(NC(=O)CCC3CC3(F)F)C2)ccccc1C1CC1 C1(C(=O)NC2CN(C(C3C(C)(C)C3C(F)F)=O)C2)CCC2(CCCC2)C1 C1(C)(CCC(=O)NC2C(NC(CC(C)OCC)=O)CCC2)CCC(=O)N1 C(=O)(C(C(c1ccccc1)N(C)C)N1CC(C)(OC)C1)NCCOC N1(C(C(C)OC(C)=O)=O)CCC(C(=O)N(C2CC2)CC2CCCO2)CC1 c1(C(=O)NCC(C)(C)CNC(=O)CC2CC3CCC2O3)c[nH]c2c(Cl)cccc12 c1(C(=O)NCC(=C)CCNC(=O)C(C2CCC(=O)N2)C)ccc(OC)cc1 N1(C(CC(C)(C)O)=O)CC(c2cn(-c3cccc(F)c3F)nn2)C(C)(C)C1 C(C#Cc1cccnc1)NC(CC(C)N(C(C(C)N=[N+]=[N-])=O)C)=O c1(NC(C(C)OCCC2CN(C(=O)CCN(C3CCCC3)C)C2)=O)ccncc1 n1(CCOC)ccc(C(=O)NCC2CCCN2C(=O)CC2(O)CCOC2)n1 c1(N2C3C(NCc4cccc(OC)c4)C(C3)C2)ccnc2ccnn12 N1(C(Cn2c(C)csc2=O)=O)CCCCC1C1CCCN1c1ccnc(Cl)n1 c1(C(C(=O)N(C2CN(C(C(CC(C)C)O)=O)C2)C)C)ccc([N+](=O)[O-])cc1 CC1C(NC(=O)CCNC(c2c[nH]c(=N)s2)=O)CCCN1C(c1ccccc1)=O c1(C(=O)NC2(CC)CCN(C(CCCC#C)=O)CC2)cc(F)c(F)c(F)c1F C(=O)(C1=CCCC1(C)C)NC12C(CN(C(C(CC(C)C)NC(N)=O)=O)C1)CC2 C1(NC(c2cccc(C3CC3)n2)=O)CCCCN(C(c2n[nH]cc2Cl)=O)CC1 c1(C(N(CCC(C(C)C)NC(=O)CN2CCCS2(=O)=O)C)=O)nccc(Cl)c1F CC1(C)CCCC1C(=O)NCCC1CCN(C(C2(C(N)=O)CC2)=O)C1 C(=O)(CS(=O)(=O)NC)NCC(CCSC)NC(=O)CCCNC1CC1 C1(CN(C(=O)C(F)C2CCOC2)C)CCC(CNC(C23CC2CNC3=O)=O)CC1 C(=O)(CC(C)CC(=O)OC)N1CCC(C=CC(NOCC2CC(=C)C2)=O)CC1 C(=O)(C1CCCc2ccnn21)NC1CCCCN(c2snc(COC)n2)C1 N1(C(c2cc(OC)n[nH]2)=O)CC(O)CCC1C(N1CC(n2cccn2)C1)=O CCC(CC(=O)NC1(CCCNC(c2cc(CC(C)C)[nH]n2)=O)CC1)C(F)F N1(C(C(C(=O)OC)C)=O)CCN(C(C)=O)C2CC12.C1C(=O)N1CC(C)C C1(CNC(C(C)OC2COC2)=O)CCN(C(c2c(Cl)cnn2C)=O)C12CC2 C1(NC(Cc2cccc(C(C)(C)C)c2)=O)CCCCN(c2ncnc(=N)[nH]2)C1 c1(NC(C(C(C)C)NC(CCC(C)SC)=O)=O)c(C)cccc1C c1(C(=O)NCC2OCCN(CC(=O)OC)C2)cc(Br)c(OC)cc1OC c1(OC)c[nH]c(C(N2CCC(CNC(=O)Cn3ccc(C)n3)C2(C)C)=O)cc1=O C=CC1(CC(=O)NCCCCCN(C)C(c2conc2C)=O)CCC1 Cc1[nH]nc(C(N2CC(NC(=O)C(c3c(C)noc3C)C)C(O)C2)=O)c1C C1(C(=O)NC2(CCNC(c3c(CC)n[nH]c3)=O)CCC2)CC(C)OC(C)C1 N1(C(CCCOCC)=O)CCSCC1CCNC(c1cccc(F)c1)=O C1(CNC(c2cc(-c3ccccc3)ns2)=O)CC(O)CN1C(c1csc(O)n1)=O N1(C(CCC=CC)=O)CCCC2(C1)CN(C(=O)C(C)S)CCO2 C1(CC(N2CCC(CCCNC(CCCOC)=O)CC2)=O)CCCCC1(C)C c1(C(=O)NC(C(=O)NC(CC#C)CO)C2(O)CCC2)cc(C)cc(C#N)c1 C1(OC)CN(C(c2sc(C3CC3)nc2C)=O)CC1NC(=O)C(C)(C)c1cscn1 N1(C(CC(C)OC)=O)CCC2(CC1)CC(N=c1nc(C(F)(F)F)[nH]s1)CCO2 c1(C(=O)Nc2cn(C)nc2C(F)F)cncc2c(Br)cccc12 C(=O)(CCCC(OC)OC)NCC(C(=O)NC(CC)Cn1cncn1)CC1CC1 N1(C(C(n2cc(Cl)cn2)C)=O)CC(CNC(=O)CN2CCOCC2)CC1(C)C C=CC(C)(CC)C(=O)NC(C)CC1CN(C(c2ccc(-c3ccncc3)s2)=O)C1 CC(C)C(C(C)NC(=O)C=C1CCOCC1)NC(=O)C(N)=O N1(C(C2N(C(c3c(COC)cccc3)=O)CCC2)=O)CC(=O)N(C)CC1C Cc1cc(C(=O)NC(C)CC(C)NC(c2ncccc2NS(C)(=O)=O)=O)[nH]c1C c1(C(N2CC(CC(C)NC(C3CCC3)=O)C2)=O)cnn2c1OCC(F)C2 C1(NC(C23C(CN(C(c4cnc(C)s4)=O)C2)C3)=O)CCCOC12CCC2 CCC(C)CCC(=O)NCC1CC(NC(c2cc(=N)[nH]cc2Br)=O)C1 CCCCC(F)C(=O)NCC1C(C(=O)NCC2(CC3CC3)CC2)C1(C)C C1(NC(C2(COC)CCC2)=O)COC2(C1)CN(C(=O)C(C)CS(C)(=O)=O)C2 CC1(C)CCC(CCNC(C2CC(O)CN2C(C2COC(=O)N2)=O)=O)O1 Cc1cccc(O)c1C(=O)NCC(O)CNC(c1cnc(N)cn1)=O c1(C(=O)NC2(CO)CCCN(C(=O)CCC3CCC3)C2)cc(F)c2[nH]nnc2c1 N1(C(COC)=O)CC(C)(C)CCC1CNC(=O)C(O)Cc1cccc(OC)c1 c1(C(=O)Nc2cc(C)c(C(=O)N(C)C)cc2)ncnc2c1OCCO2 Cc1cc(C(=O)NC(C2(O)CN(C(=O)Cc3ccon3)C2)C)ccc1Cl Cc1cc(C(=O)NCC2CCN2C(C2CC(C)C2)=O)n(CC(F)F)n1 c1(CN2CC(CC)OCC2)nc2c(c(=NCc3c(C)noc3C)[nH]1)CSC2 C1(NC(=O)OC(C)(C)C)COCC1NCCCn1cc(-c2ccccc2)cn1 c1(C(=O)NCC2C(CNC(c3cnc(C(C)=O)s3)=O)C2)cc(C(F)F)ccc1F CC1CCCCC1(CNC(c1nnn(C)n1)=O)NC(=O)CC(C)CN(C)C c1(C(=O)NC2(CC(=O)Nc3cnn(-c4ccncc4)c3)CC2)ccc([N+](=O)[O-])o1 C(CCC#C)(C(=O)NC(C)(C)C)N(CC#C)C CCCC(CC)C(=O)NC(c1nocc1C(=O)NCC1(C)COCCO1)C Cc1nc(O)[nH]c1C(=O)NCC1CCCCN1C(C1C(C)C1(F)F)=O c1(NC(c2n(C)cc(Nc3nc(OC)cc(OC)n3)n2)=O)cc(C)c(C)cc1Br C(=O)(CCC(=O)N(C(COCC)C(=O)N(C)CCO)C)NCCC C1(CC)CN(C(=O)CCC(=O)N(C)C)CCN1C(=O)C(=CC1CCCCCC1)C C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1C2(CCN(C(c3ccc(CSC)o3)=O)C2)C1 c1(OC)ccc(C(N2CCC(C(=O)NCC3(CN=[N+]=[N-])CC3)C2CC)=O)cc1 C1(C(=O)NCCC2CCN(C(=O)C(C)OCC(F)(F)F)CC2)(CC)CC(C)(C)C1 N1(C(c2c(OC)cnc(Cl)c2)=O)CCC(C2CC2NC(C2CC2F)=O)CC1 C1(CNC(C=CCC)=O)C(CC)CCN1C(C1CCCNC1=O)=O N1(C(C(C)CC(F)F)=O)CCC2(CC(C(N3CCC(c4cc[nH]n4)C3)=O)C2)C1 N1(C(C)=O)CCC(C)CC1C(C1(F)CCCCC1)=O N1(c2n(Cc3c(Cl)cc(F)c(F)c3F)nnn2)CCCC(C2CCNCC2)C1 N1(C(c2c(CC)occ2)=O)CC2CC(C(=O)N(CCCN(C)C)CC)(C2)C1 Fc1ccc(C2CCC(n3cc(-c4nc(C(F)(F)F)cs4)nn3)C2)cc1F c1(C(=O)NCC2C3CN(C(C(CC=C)CC)=O)CC32)nc2cnccc2s1 CC1=C(C(=O)NC2CC(C)(NC(c3cnn(CC(F)(F)F)n3)=O)C2)CCO1 CC1CCCC(CCNC(=O)NCc2cccc(C3CC3)n2)O1 C1(C)(CNC(CC2(C)CC(NC(C=CC(=O)N(C)C)=O)C2)=O)CCCCC1 c1(NC(C2N(C(Cc3c(CC)con3)=O)CCC2CC)=O)cc(C)cc(C)c1O C1(CNC(c2scc(C(C)=O)c2)=O)C(C)CCN1C(=O)Cc1ncccc1F Cc1nc(C)c(CNC(C2COCCN2C(=O)C(C)O)=O)s1 c1(N2C(C)(C(=O)Nc3cnoc3)CCC2)ccn2ncc(I)c2n1 CC1CCC(C(=O)NCC(C2CC2)NC(c2csc(C(F)(F)F)n2)=O)CC1 c1(C(N2CC(C)N(C(C3CC(C4CC4)C3)=O)CC2)=O)c[nH]c2ncccc12 N(C(=NCCF)N1CCCC(c2ccccn2)C1)C(C=C)C C1(CNC(C2C(OC)CCC2)=O)CC2(CC(NC(c3cnc(C4CC4)o3)=O)C2)C1 Cc1[nH]c2ncccc2c1C(=O)NCCNC(=O)C(CC=CCl)c1ccccc1 CC(F)(F)CCC(=O)NCCOCC(=O)NCCCF N1(C(C(C)SC(F)(F)F)=O)CC(NC(c2cccc(N)c2O)=O)CC(C)(C)C1 C1(C(=O)NCC2(N(C)C)CC2)CN(C(=O)CC2CCC2)CC1C(F)F C(C)(N=c1[nH]c2c(c(=NCCN(CC(F)F)C)[nH]1)SCC2)c1ccc(C)o1 C1(NC(C(C=CC)O)=O)CCN(C(c2cscc2Cl)=O)C1c1ccccc1 C(=O)(C1CCCn2cnnc21)NCCC(C)NC(c1c(=O)n(C)nc(C)c1C)=O c1(NC(C2CC(O)(CNC(c3ccn(C(C)C)c3)=O)C2)=O)cn(C)c(=O)nc1O C1(C(=O)NC2CC(C)N(C(=O)Cn3cnnc3O)CC2)C2CCC1(C)C2(C)C c1(C(N2CCC(CNC(C=CCOC)=O)(OC)C2)=O)cn2ccccc2n1 C1(N(C(CCN(C)CC)=O)CC)CCCN(C(=O)C(O)c2ccsc2)C1 C(=O)(C1=CC2CCC(C1)C2)NCC1CN(C(C2CCOC2)=O)CC(C)(C)O1 CCC(CC(=O)NC(CC(F)F)C(=O)NCC(CC)C(C)C)C(C)C c1(C(N(CC(N2CCN(C(CCC(C)C)=O)CC2)=O)C)=O)c(N)ccc(F)c1F CCCC(CNC(=O)Cn1cncn1)NC(c1cccs1)=O C=CCC(C)(CC)C(=O)NCC(O)CCNC(c1ccnc(Cl)c1O)=O C#Cc1cnn(CC(=O)N(C(C)CNC(=O)CN2CCC(C)(C)C2)C)c1 C(=O)(C(C)C(C)(C)C)NCC1(CNC(CCC#C)=O)CCCC1 C1(CCC)CN(C(=O)COc2cc(C)on2)CC1NC(c1sc(F)cc1C)=O C1(CC(N2C(CNC(c3c(C)cc(CO)o3)=O)CCC2)=O)CCC(C)(C)CO1 Cc1nc2c(cnn2C(C)C)cc1C(N1CCC(n2cc(C(C)(C)CO)nn2)C1)=O c1(C(C)(C)C)ccc(C(=O)NCC(C)(O)CNC(=O)C(F)C2CC2)cc1Cl C1(NC(CSCCC(C)C)=O)COCC1NC(=O)C(F)CC1CC1 c1(C(=O)NC(CC=C)CNC(C2C(C(F)F)C2(C)C)=O)ccn(CC)c1C C(C)(C)(CCC(=O)N1CCCC(O)C1C)NC(CC=CC)=O Cc1nn(C)c(C(F)F)c1C(=O)NCCC(C)(C)NC(=O)C=CC1CCCN1C c1(OC)cc(CNN(C)C)cc(Br)c1.C1(C)(CO)CCCC1 c1(OC)cc(CC(=O)NC(C2CN(C(=O)CN3CSCC3=O)C2)C)ccn1 C(=O)(C(C)CC(F)F)NCC(CC(C)C)NC(c1c(C)oc(-c2ccsc2)c1)=O N1(C(CCCOCCOC)=O)CCC(F)(C(=O)NCc2conc2C2CC2)C1.CN C1Cn2ccnc2NC1=O.C1(NC(=O)OC(C)(C)C)(CO)CC(O)C1 c1(C(=O)NCC(CNC(C2CCN(C(C)C)CC2)=O)CO)cccc2scnc12 C1(O)(CN(C)C(c2cc(Cl)nn2C)=O)CCN(C(C2(C)COC(=O)N2)=O)C1 N1(CC(CCCC)=O)CC2(NC(=O)OC(C)(C)C)CCC2(C(=O)OC)C1 Cc1ccc(C(=O)OC2CCOC(C)(C)C2)c(O)n1 C1(C2CCCN(C(C3CC3Cc3cccnc3)=O)C2)(NC(=O)C=CC2CCC2)CC1 n1(C(C)C)cc(CN(C(C)C(C)C)C(=O)CC2(C)CC2)c(O)nc1=O C(=O)(C1=COCCC1)NCc1c(N)cncc1.C12CCC1C(=O)N2 c1(OC)ccc(C(c2nnnn2C2CC(F)(F)C2)NC2CC23CCC3)c(F)c1 N1(C(c2c(C)c[nH]c2)=O)CC(CNC(c2nnc(C)n2C)=O)C(C)(C)C1 N1(C(N(CCCSC)C)=O)CCC(CN)C(C)C1 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CN(C(c1ccc(C(C)O)cc1)=O)C2 O=C(CCCCC(F)(F)F)NCCC1CN(C(C2CCC(F)(F)C2)=O)C1 CC(CC(C)(F)F)C(=O)N1CC2CC2(NC(c2ccnc(N(C)C)c2)=O)C1 C1(NC(c2ccc(OC)cc2)c2n(C(CC)(C)C)nnn2)CCC=CCCC1 c1(C(=O)NCC2(NC(CN(C(C)=O)C)=O)COC2)cn(C2COCC2F)nn1 c1(C(=O)NCCN(CCOC)C(C2C3COCC23)=O)csnc1OC c1(NC(C2C=CCN2Cc2ccc(Br)cc2O)=O)cc(F)c(F)c(Cl)c1Br C1(C(=O)NCCC2(OC)CN(C(C3CCNC3=O)=O)C2)CCCN(S(N)(=O)=O)C1 c1(OCC)ccccc1NC(C)CNC(c1cc(C)n(C(C)CC)n1)=O N1(C(Cn2nnc(C)n2)=O)CCC(CNC(C2(CCF)CCOCC2)=O)C(C)C1 C12(NC(c3scc(C)c3)=O)CCCC1N(C(c1cc(C(F)F)ccn1)=O)CCC2 C(=O)(C(C)C(C)COC)NCC(CCOC)NC(C(CC=CCC)C)=O C(=O)(C(CC(C)C)N(C(=O)CCCNC(=O)N(C)C)C)NCC(=O)OC N1(CCCNC(CCN(C(CC)CC)C)=O)CCC(NC(C2CCCCS2)=O)C1 c1(C(C)(C)C(=O)NC(=O)CNC(C2CNC2)(C)C)ccc(F)c(F)c1 C(C)(C(N=c1ccnc(C2CC2)[nH]1)C(C)C)NC(c1c(CC)nco1)=O C=CCC(F)(F)CNC(=O)C(CC1CCOCC1)NC(=O)C(c1ccn(C)n1)C N1(C(C2(CCC)CC2)=O)CC(NC(C2CCC(F)(F)C2)=O)C(C(F)F)C1 c1(C(=O)NC2CC(C)(CNC(c3cc(=O)cc(Cl)[nH]3)=O)C2)ccc(C#N)c(F)c1 Cc1c(CNC(=O)NC(C)(CO)CC(C)C)cccc1C(F)(F)F C1(C(=O)NCc2onc(C)n2)C2CCC(C2)N1C(C1C2CCCCCC12)=O C(=O)(C(CO)C(C)(C)C)N1C2CC(C(N3CC4(CN(C(C)=O)C4)C3)=O)C1CC2 Cc1cc(C(=O)NC(C2(O)CCN(C(C3CCSC3)=O)CC2)C)nc(C)c1 Cc1nccc(C(=O)NCCC2(C)CCN(C(=O)C(CC(C)C)N(C)C)C2)c1O C1(C(N2CCCCC(N(C(CCCSC)=O)C)C2)=O)CCCCCC1(F)F c1(C(=O)NCC2CCN(C(CCNC(=O)NC)=O)C2)nccc(C)c1O CC(=O)CCC(=O)NC1CC(CCC(N2CC3CC3C2)=O)C1 N1(C(C(C)OCC)=O)CC2(CCN(C(C3CC(F)C(=O)N3)=O)CC2)C1 c1(C(N(CCCCNC(=O)C=Cc2cncs2)C)=O)c(O)cccc1F c1(C(N2CCC3CC23C(=O)NC(CO)C2(O)CC2)=O)cccc(O)c1F C1(CC)CN(C(=O)NCC2CCCOC2C(C)(C)C)CCN(C)C1 CC1CCc2ncc(C(=O)N(C)CC3COCCN3C(=O)CC3OCCO3)n2C1 Cc1cn2ccnc(C(N3CCC(C)C(NC(C4CCC(C)CC4)=O)C3)=O)c2n1 C12(NC(c3nc(CC)sc3N)=O)CCCC1CN(C(=O)C(O)c1cnc[nH]1)C2 CCC(CC)CC(F)C(=O)N1CCC(F)(CNC(c2cn(C3CCC3)nn2)=O)C1 N1(C(C(COCC)(C)C)=O)CC(C(N2CCC3C(C(=O)OC)C3C2)=O)CCC1C C1(C(N2CC(C(N)=O)(CNC(c3ccc(CC)cn3)=O)C2)=O)CC2C(C1)C2(C)C C(CCOCCO)(C(=O)Nc1ncccc1CO)NC(C(C)NC(=O)NC)=O CC(CS(C)(=O)=O)C(=O)NC1CCC12CN(C(c1cccn3cncc13)=O)C2 c1(NCCNC(C2C(CCCC)CCC2)=O)ccc(Br)c(C)c1[N+](=O)[O-] c1(C(=O)OC)c(Cl)nc[nH]c1=NCC12CC1CN(C(c1cc(C)nc(C)c1)=O)C2 c1(CC)ncc(C(=O)NC2CCC(CC(=O)NCc3ccco3)CC2)cn1 c1(OCC)oc(C(F)(F)F)nc1C(=O)NCC1(Cn2cc(CCSC)nn2)CC1 C(N=c1nc2c(cnn2C)c(NCc2coc(C)c2)[nH]1)C1C(C(=C)C)OCC1 C1(F)(C(N(CC(C2CC2)OC)C)=O)CCCN(C(=O)C=C(C)C)C1 N1(c2ncc(C(=O)OC)c(C)c2)CCC(C2CC2)C1CNC(C1CC1C)=O C(=O)(C1CCCc2cncn21)NC(C(C)NC(c1c(C)ncs1)=O)CO Cc1cnc(C(=O)NC2C3CN(C(=O)Cc4cccc(C#N)c4)CC23)c(Br)c1 S(=O)(=O)(c1cccnc1N1CC2(C)CSCC2(C)C1)NCc1ccc(CC)o1 C(CCCCCCC(=O)NC1CC1CNC(c1ccc(Cl)nc1O)=O)SC c1(C(=O)NC2CC(NC(c3c(C)nc(C)s3)=O)C(O)C2)ccc(F)c(N)c1 N1(c2nc(OCC)c(C)cn2)C2CCCC1CN(C(=O)C(C)(C)CC(F)F)C2 C12C3CCC(C3)C1C(=O)N2.c1(C(N(C(C)CN(C)C)CC)=O)ccns1 C1(CN(C)CCNC(C2(CC)C(COC)NC2=O)=O)Cc2ccccc2C1(C)C O=S(=O)(c1ccc(NCC2CC2(F)F)c(Br)c1)N(C1CCCO1)Cc1ncccn1 n1(C(CC)CC)cc(-c2ccc(SCC3CCS(=O)(=O)C3)cc2)c(C)n1 N(C(=NCCC(=O)NCC1CCOC1)NCC(F)(F)C(F)F)C1CCS(=O)(=O)C1 c1(N(CC(C)(C)C)C)[nH]c(=NCCC(C)c2ccccc2)nc2scnc12 CC1CC(NC(c2cc(N)ccc2Cl)=O)CCN1C(c1cc(C(F)F)ncn1)=O c1(C(=O)NC(C)C(C)NC(c2ccc(O)s2)=O)cc2n(n1)CCNC2=O C#CCCN=C(NCCS(=O)(=O)CC)NCC1COCCO1 C12(CN(C(CC(C)(C)N(C(Cc3c(C)ccnc3)=O)C)=O)CC)CCCC1CCO2 C(=O)(CC(C)(C)C(F)F)NC1(CSC)CCC1.C(C1C(=O)N1)NS(C)(=O)=O c1(CC(C(=O)N(C(C)CCNC(=O)Cc2ccco2)C)C)ccc(Cl)cc1 c1(C(=O)NCC23CC(NC(C(C(C)(C)C)=O)=O)(C2)C3)ccnc2ccsc12 C1(NC(=O)CC2(C(F)(F)F)CC2)CC(NC(C2CCCCC2)=O)C12CCOCC2 C(c1ccccc1OC)=C(C(=O)NC(CC)CNC(C1CC1CC)=O)C C(=O)(C1CCc2ccccc21)N1C(C)CC(CC(=O)NCCC(C)(C)CO)C1 C(C(C)N=c1nc(SC)[nH]s1)N(C(c1c(OC)nsc1)=O)C c1(C(N(CCNC(=O)C(F)=C2CCC2)C2CC2)=O)cn(-c2ncccn2)cn1 c1(C(=O)NCCOCCNC(c2c(C)oc(Cl)n2)=O)cc2c([nH]1)CCOC2 C1(NC(c2n(CC)ncc2)=O)CN(C(=O)Cn2cc(C)ccc2=O)CCC1C c1(COC)cc(F)ccc1C(c1cccc(C(N2CCC(C(=O)OC)C2)=O)c1)=O C1(CCOC(C2N(CC)CCCC2)=O)CCC2(CCOCC2)O1 C1(N(C)C(c2cc(Br)co2)=O)CN(C(=O)CCc2cn(C)nn2)CC1(C)C Cc1cc2cc(C(N3CCN(C)CC3C(=O)O)=O)ccc2s1 c1(OC)ccc(-c2n[nH]c(CN(C(=O)CCc3ccnc(Cl)c3)CC(C)O)n2)cc1 c1(CN2CC(NC(c3cnc(C(C)(C)C)nc3)=O)C2)c(O)ccc2ccccc12 C(=O)(C1=C(Cl)CCOC1)NCCCOCCNC(C1C(C)(C)C(F)(F)C1)=O S(=O)(=O)(C1CN(C(N(C)Cc2ccccc2)=O)C1)NCCn1cnnc1 C(=O)(C1=C(C)CCCC1)NC1CCN(c2cc(CC)nc(C)n2)C(C)C1 c1(C2(C(=O)NCC3CCN3C(=O)CCCNc3ccsn3)CC2)ccc(F)cc1 N1(C(C(CCC)NC(N)=O)=O)CCC(C(=O)N(C)CCNC(C)=O)C(C)(C)C1 CC(C)C(C)(CNC1(N2CCOCC2)CCSC1)NC(=O)OC(C)(C)C c1(OC)cccc(CNC(=O)C=CC(C)NC(=O)Cc2sccc2Cl)c1 C1(NC(C2CCS(=O)CC2)=O)CCN(C(C2CCc3nccn3C2)=O)C12CCC2 CCC(C)(O)C(=O)NC1CC(C(=O)NCC(=O)NCC(F)F)C1 C(c1ccc2occc2c1)=CC(N1CCC(C(C)NC(c2ccns2)=O)CC1)=O c1(CN2CCC3(C(C(=O)NC(c4ccccc4Br)C)C3)C2)cc(Br)c(F)cc1O n1(-c2cc(OC)ncc2)ccc2ccc(CN3CCc4nc(CO)cn4C3)cc12 c1(C(=O)NCCC2(O)CN(C(CCC(=C)Br)=O)C2)ccc(N(C)C)cc1F C1(C(C)NC(=O)Cn2cnnn2)CN(C(c2cnc(C(F)(F)F)cn2)=O)CCO1 C1(N(C(C(CC)C)=O)CCO)CCN(C(C2CC2F)=O)CC1 c1(C2N(C(C3CCC(NC(c4c(C)nc[nH]4)=O)CC3)=O)CCC2)cc(F)cc(Cl)c1 c1(OC)cc(C(=O)NC2CC2NC(=O)C(c2ccccn2)O)on1 CS(=O)C1CN(C(C2CCOCC2NC(=O)Cc2noc(C3CC3)n2)=O)C1 c1(C(N(C2CCN(C(CC3CC(SC)C3)=O)CC2)C)=O)ccc(C(C)C)c(F)c1 CC(C)CC(=O)C(=O)N1CCC(C)(NC(C2CC2(C)Br)=O)CC1 CP(C)(=O)C1CCC=C1C(=O)NCC1CCCN1C(=O)Cc1cnoc1 C(CCC(=O)N(CCn1ccnc1)C(C)C)(C(C)C)NC(CSCCC)=O C(CC(C)(C)C)(C(=O)NC1CCN(C(=O)C(C2CC2)C2CC2)CC1O)OC N1(C(CCNCC)=O)CCCC12CCCC2.C(=O)(C(C(=O)OC)OC(C)C1CC1)N C1(CNC(C2(OC)CCCC2)=O)COCCN1C(c1cc(Br)c(C)s1)=O CC12CC1CCN2C(C1CCC(NC(c2ncccc2Cl)=O)C1)=O c1(C(N2CCC(N(C(C3CC3(Cl)Cl)=O)CC)C2)=O)cc(OC)cc(F)c1 c1(OC)ccc(Cl)c(C(N2CCCCC2CNC(c2ccc(C)c(F)c2)=O)=O)n1 C1(C(=O)NC(CN(C)C(c2cnn3c2OCC3)=O)(C)C)CCc2ccccc2O1 C1(C)(CNC(c2c(CC)n(CC)nn2)=O)CC(OC)CN1C(=O)CC(C)C N1(C(c2ccc(CCC)s2)=O)CCC(C(C)(C)C)(CNC(c2c[nH]nc2C)=O)C1 CC1COCC(C)N1C(C1CCOC(C)(C)C1)=O C1(NC(C(C)(C)SCC)=O)CCCN(C(=O)CCOC2CC2)C1 C(CC(C)(C)C)COC(C(=O)NC(CC=CC(=O)OC)(C)C)C c1(C2C(C(=O)NCCN(C(C3(CC#C)CC3)=O)CCOCCO)C2)ccncc1 C12(C(=O)NC3(CNC(c4nn(C)c(C5CC5)c4)=O)CC3)CCC(C1)C(C)(C)O2 c1(N2CC(F)(C(=O)NC(c3ccc(Cl)cc3Cl)C)C2)ccn2ncc(Br)c2n1 C(=O)(CCCCCS(N)(=O)=O)NCC(=O)N(C1CCN(C(C)=O)CC1)CCCC C1(N(C)C(c2cccs2)=O)CN(C(c2c(C(F)(F)F)cnn2C)=O)CC1O CC1CN(C(=O)CCCN(C)C(c2cn(C)cn2)=O)CC1C(N)=O c1(CC(=O)NCC2N(C(c3nc(CC)oc3C)=O)CC(O)C2)ccc(F)c(Cl)c1 CC(C)(C)CC(O)C(=O)NCC1(O)CCN(C(C2CC(n3ccnn3)C2)=O)CC1 C(=O)(C(C(C)C)N(C)C)NC(COC)C(=O)NCC1CCOC1C c1(C(=O)NCC(C)(O)CNC(=O)C=CBr)cc2cscc2s1 N1(C(c2c(C)ncc(Cl)c2)=O)CC2COCCC2(NC(=O)CN(S(C)(=O)=O)C)C1 N1(C(C=CC)=O)CCC(C(=O)NCC(O)CCC2CC2)C(O)C1 CCCCC(O)C(=O)NCC#CCNC(C1COCCN1C)=O N1(C(C(CSC)O)=O)CCCC2(C1)CN(C(c1cc(C)n(C3CC3)c1C)=O)C2 c12nc(-c3ccc(Cl)cc3)nn1C2C1(C)CC1.N(C)(C)CC N1(C(c2ccc(C(C)=O)cc2CC)=O)CCC2CN(C(C34CCC3CC4)=O)CC12 Cc1nc2cccc(C(=O)Nc3nc4c(s3)CCC4)n2n1 N1(C(c2c(C)cc(C)s2)=O)CCCC(C)(C)C1CNC(C12CCCC(CO1)C2)=O N1(C(C2(C)CC2)=O)CCN(C(C2CC2Sc2ccccc2)=O)CC(O)C1 c1(C(=O)NCC2CCCN2C(C2CC=CC2)=O)cc2cc(Cl)ccc2o1 c1(C(=O)NC2CCCN(C(C3(C=C)CC3)=O)C2)ccc(N)c(C)c1F C(CCC)(C(O)C(=O)NCC1(Cl)CC1(F)F)NC(COC1(C#C)COC1)=O CCCCC(C(=O)NCC(C)CN(C)C(c1csc(CCC)n1)=O)N(C)C C(CCC(C)C(=O)NCC1CC2(CC2)CN1C(c1cc(N)cc(N)c1)=O)OC c1(C(=O)NCC=CCNC(CCCCN(C)C)=O)nn2cccnc2c1Cl c1(NC(C2(O)CCN(C(c3nccnc3N)=O)CC2)C)ncc2ncnc-2[nH]1 CC1=NOC2(CCN(C(=O)NC3CCC4(CCCCC4)O3)CC2)C1 Cc1ccc2cc(C(=O)NCCOC(=O)C3CC3)cnc2c1 c1(C(N2C(CNC(CCCCC=C)=O)COCC2)=O)cc2c(cnn2C)nc1O N1(C(C2(OCC)CCCC2)=O)CCC(OCCCNC(c2ccsn2)=O)CC1 CC1CCC(O)(C(=O)NCC2(F)CCC(NC(c3ccnc(CO)c3)=O)C2)CC1 c1(C(N2CC(O)(CNC(=O)COCC3CCCO3)C2)=O)cnc(O)c(Br)c1 N1(C(C2(OC(C)C)CCC2)=O)CC(n2cc(Cc3ccc(F)cc3)nn2)C(C)C1 CCC(N=c1ccnc(COC(N2CCCCC2C)=O)[nH]1)c1cc(OC)ccn1 C=CC1(C(=O)NCC2(CNC(=O)CC3CCOC(C)(C)C3)CCC2)CCOCC1 c1(COC(=O)CSC2CN(C(=O)CCC(=O)N3CCOCC3)C2)ccccc1O N1(C(CC(C(=O)OC)C)=O)CCCC12CCN(C(C1CN3CCCN1CC3)=O)C2 c1(C(N(C)Cc2cn(CCOC3CCOC3)nn2)=O)c[nH]c2cccc(F)c12 N1(C(CCCCOC(C)C)=O)CCC(NC(c2cc(C3CC3C)on2)=O)C(O)C1 C(=O)(C(C)(CO)NC(c1cncc(OCC)c1)=O)NC1(OCC)CC1 c1(OC)cccc([N+](=O)[O-])c1C(N1CC(NC(c2cncs2)=O)C(C#N)C1)=O c1(-c2n(C(CC#C)C3CC3)c(N3CC=C(C)C3)nn2)nc2cc(C)ccc2o1 Cc1cc(C(=O)NCc2cn(C3CN(C(C4CC45CCOC5)=O)C3)nn2)n(C)n1 S(=O)(=O)(c1c(F)cccc1F)N1CCC(F)(C(=O)Nc2c(I)ccc(C#N)c2)C1 C1(NC(COC)=O)CN(C(c2sccc2F)=O)CC2(CC2)C1 c1(C(=O)NC2CC(NC(C3C(c4nc(C)[nH]n4)C3(C)C)=O)C2)cnccc1C c1(NCC(=O)NC(C)CN(C)C(c2csc(O)n2)=O)ccc(C(F)(F)F)cn1 c1(CC(=O)N(CCN(C(COCC(=O)OC)=O)C)C)cnc2n1CCCC2C C1(NC(c2ccc(C(F)F)cn2)=O)CCN(C(C2CCCCS2)=O)C12CCCC2 N1(C(CC(CC)C)=O)CCC(F)C(NC(=O)CCOCc2ccccc2)C1 N1(C(C(N2CCCCC2)C)=O)C(CNC(=O)CCCCc2cnn[nH]2)CC2CC12 C1(O)(CN(C(C(COC)(C)OC)=O)C)CCCN(C(=O)C(=Cc2cnc[nH]2)C)C1 N1(C(C(NOC)=O)=O)CC(=O)NC2CN(C(c3cnn(C(C)(C)C)c3)=O)CCC12 c1(C(=O)NCC2(C)CCN(C(C3C(CC)C3)=O)C2)cc(O)c2c(cnn2C)c1 CCCCCCC(C)CC(=O)N1CCN(C(=O)CNC(=O)OC)CC1CC C(=O)(C1=CC(C)(CC)C1)N(CCNC(C1(C(F)(F)F)CC(=C)C1)=O)CC1CC1 Cn1nc(CNC(C2CC(OC)C2)=O)cc1C(=O)NC(CO)CCC1CC1 c1(OC)ccccc1OCC1(OCc2cnc(C(=O)O)s2)CC1 N1(C(Cc2cc(C)sc2)=O)CCCC(C(=O)NCc2cc(C3CC3)no2)C1.CN C1(NC(c2cc(Cl)cc(F)c2F)=O)COC2(CCN(C(=O)COC3CCC3)C2)C1 C1(C#N)(C(N2CCCC(Cc3onc(C)n3)C2C)=O)CCS(=O)(=O)CC1 Cc1nc2ccccn2c1C(N1CC2CC2(CNC(=O)CCc2ncco2)C1)=O c1(OC)cc(OC)c(C(=O)NCCCCCCNC(C2(O)COC2)=O)c(OC)c1 N=c1ccc(C(=O)NCC2CCCN(C(C3(c4ncc(Br)cn4)CC3)=O)C2)n[nH]1 c1(C(N2CC(CNC(c3c(OC)ccc(Br)c3)=O)C2)=O)ccc(F)c(Cl)c1C c1(NC(C(C2(O)CCC2)NC(Cc2ccc(C)nc2)=O)=O)cnc(C)nc1C C(CCCCC(=O)NCC1CCCOCC1)N(C)C(c1cc(O)cs1)=O c1(C(N)=O)cc(CC(N2CC(CCNC(=O)CC3CC3C)C2)=O)ccn1 c1(C(=O)NCC2(F)CC(CNC(C34CSCC3C4)=O)C2)c[nH]c2nc(Cl)ccc12 CC(C)C(CCN(C)C(C1CCC(F)(F)C1)=O)NC(C1CCCN1C=O)=O C1(C(N2CC(C)C2C(=O)N(CC(C)(C)CN(C)C)C)=O)CCCN(C)C1 c1(N(C(C)C)C)[nH]c(=NCC(C2CC2)C2CC2)nc2ncn(C)c12.C1(=O)CN1 C1(C(=O)NC2C=CCN(C(C3CCC(=O)C3)=O)C2)CCc2ccccc2C1 C1(C(N2CC(COC)(CNC(C3CC(F)(F)C3)=O)C2)=O)CN2CCC1(C)CC2 C1(NC(c2c(C)noc2C)CC(=O)NCC(=O)OCC)CCc2n[nH]cc2C1.OCC N1(C(C2CC(C)(F)C2)=O)CCCC(F)(CNC(C2CCC3CCC2O3)=O)C1 C12(NC(=O)C=CCO)CCCC1CN(C(c1cccn1C1CCC1)=O)C2 C(C)(CCCCCO)NC(C(Cn1ccnn1)NC(CSCCOC)=O)=O N1(C(c2cccc(N=[N+]=[N-])c2)=O)CC2CCCC2(NC(=O)Cc2nncs2)C1 C#Cc1ccc(CC(=O)N(C(C)CCNC(=O)CC2CCC(C)(C)O2)C)cc1 CCCC(C)S(=O)(=O)NC(c1ccnn1-c1cccnc1)=O c1(CC(=O)NCC(C)NC(C(CCC)C#N)=O)cc(Cl)c2c(c1)OCCCO2 c1(CNC2CC(NC(c3cc(Cl)c(Cl)c(Cl)c3)=O)C2)ccc(F)c(F)c1F c1(Cc2nc(C3N(C)CCOC3)on2)nc2c(s1)COCC2 c1(C(=O)OCCCC=CC(C)C)cc(N2CCCC2)cc(Br)c1 c1(C(=O)NC(CCCC)CNC(=O)C(C2CCCCC2)O)cc2cn[nH]c2cn1 C1(CCC)CN(C(=O)CCC2CCCC2)CC1C(=O)NC(c1ccco1)CO O=C1NCCN(C(=O)NCCc2n[nH]cc2Br)C1c1ccccc1Br CC(CC(=O)N1CCC(CNC(=O)Cc2cccnc2O)CC1)C(C)(C)C C(C(O)C(=O)N1CC(O)(CN(C)C(C2(F)CCOC2)=O)C1)SC C12(CNC(c3c(C)oc(C4CC4)n3)=O)CCC(C1)N(C(=O)C(C)OCC1CC1)C2 N1(C(c2c(C)cc(C)o2)=O)CC(CNC(=O)C(C)Cn2ccnc2)C(F)(F)C1 n1(CCC(=O)NC(C)CN(C(=O)C(O)C2CCCC2)C)cc(C#N)c(O)nc1=O N1(C(CC#CC)=O)CCN(C(c2cccc(C)c2)=O)CC1CC CC1CCC(CC(=O)NC2(C)CC(C(=O)NCC(CO)C3CCC3)C2)O1 c1(OC)ccc(C(=O)NCC(CNC(=O)CCCn2ccnc2C)OC)cc1C Cn1nccc(C(=O)NC2(CO)CCN(C(=O)Cn3nnc(=N)[nH]3)CC2)c1=O CC(C)C(F)(CNC(c1ccccn1)=O)C(=O)NC1C(C)(C)C1(C)C c1(CNC(C23CC(NC(C4CCCN(C)C4)=O)(C2)C3)=O)cc(F)cc(Br)c1 c1(OC)ncc(F)cc1C(=O)Nc1ccn(-c2ccc(Cl)cc2Cl)n1 C1(C2CC2)(CNC(C=CS(C)(=O)=O)=O)CCN(C(C23CCC(CC2)C3)=O)C1 C1(CC(C(=O)N(CC(CNC=O)C)C)c2ccccc2)(CC)CCOC1.OC N1(C(C2(C)CN(C(c3c(C)scc3)=O)C2)=O)CC2C(C1C(N)=O)C2(C)C C1(NC(=O)C=Cc2ccncn2)CN(C(=O)CC2CCCO2)CCC12CCC2 S(=O)(=O)(c1cc(C)ccc1C(C)C)NC1CCCC(C=C)C1 c1(C(N2CC3C(NC(=O)COc4ccc(Cl)cc4)(C3)C2)=O)ccc(O)c(F)c1F c1(OC)cc(F)c2c(C(=O)NCCCC(C)NC(C3CCC(=O)C3)=O)n[nH]c2c1 C(CS(=O)(=O)CC(=O)NN1CCCC1C(=O)NCC12CCCN(CC1)C2)OC S(=O)(=O)(c1ccc(C(N2CCCC2(C)CNC(=O)C2=CCCC2)=O)o1)N(C)C c12ccc(nc1)[nH]2.c1(C(=O)NC2(CNC(C(OCC)C3CC3)=O)CC2)sccc1C CC1CCC(C)N(C(C2CC(N(C)C(c3cc(O)nn3C)=O)C2)=O)C1 Cc1ccc(C(N2CCCC(C)(C(=O)NCc3ccco3)C2)=O)cc1S(C)(=O)=O C1(C(N(C)CC2CCCN2C(C2CCC2)=O)=O)COc2ccc(Br)cc2O1 c1(C(=O)NC2(C)CC(NC(COC3(C#C)COC3)=O)C2)cnc2ncccc2c1 c1(OC)nc(C)ncc1C(=O)NC1COCC1NC(c1cc(Cl)cnn1)=O c1(CNC(c2c(CC)n[nH]c2)=O)ccccc1C(=O)NCCN(C1CC1)CC C1(CNC(COCCSC)=O)CC12CCN(C(c1cc(C)nn1C)=O)CC2 c1(NCCc2cnc(NC(C(CCC)C)=O)s2)c(Cl)c[nH]c2nccc1-2 c1(C(=O)NCCNC(c2c(CCC)onc2C)=O)cc(F)c2c(c1)CCC2 C#CCC(O)C(=O)NC1COCC1CNC(c1sc(C)nc1C)=O C1(NC(C2C(C)OCCO2)=O)CN(C(c2cc(Br)ccc2N)=O)CC1(C)C c1(C(=O)NCC2(O)CN(C(CCSCCCC)=O)C2)ccc2cc(O)ccc2c1 S(=O)(=O)(c1ccc(=NCCC2CSC2)[nH]c1)NC1(C)CC=CCC1 CCCCCCCc1cn(C2CCN(C(C34CCCCC3C4)=O)C2)nn1 c1(COC)nccc(=NC2CCCC23CN(C(c2cn(C(C)C)nn2)=O)C3)[nH]1 C(=O)(C1=CCCOC1)O.c1(CC(=O)NC(NC)=O)ccc(O)cc1O C1(CNC(C2CC(O)CN2Cc2ccc(C3CC3)cc2)=O)CCC(F)(F)C1 Cc1ccc(F)c(C(=O)NCc2cc3occc3s2)n1 C1(c2n(C(C)C)nnn2)(Nc2cnn(C(C)C)c2S(N)(=O)=O)CCCC2(CC2)C1 N1(C(CC2C=NN(C)C2=O)=O)CCC2CCN(C(c3cc(COC)on3)=O)CC12 C(C)(CCC(=O)NCCN1CCC(NC(=O)CCc2cc(C)no2)CC1)SC c1(C(=O)OCCCN(CCO)Cc2c(OC)cccn2)sc2nccnc2c1N c1(C(=O)NCC(C)(C2CC2)NC(C(CC(C)C)F)=O)occ2c1CCOC2 c1(SCC(N2CCOCC2CC2CCOC2)C(=O)N2CCCC2)cccc(Br)c1 C1(C)(CNC(C(C)(C)CF)=O)CCN(C(=O)CCn2cncn2)CC1 N1(C(C(CC)F)=O)CCCC(N2CCN(C(c3cc(C4(C)CC4)on3)=O)CC2)C1 c1(C(N(CCN(C(CC(C)OC)=O)C)C(C)C)=O)c(C)[nH][nH]c1=N C(c1ccc([N+](=O)[O-])s1)=CC(N1C(Cc2ccccc2)CC(C)C1)=O c1(N(CCC)CCNC(c2c(OC)cccc2C)=O)nc(OC)ccc1[N+](=O)[O-] CC(C)C(CC(=O)N=c1cc2n([nH]1)CCCC2)NC(C1(C)CNC(=O)N1)=O C1(CNC(c2cc(Cl)ns2)=O)CN(C(=O)Cn2cccnc2=O)CC2(CCC2)O1 CCCCS(=O)(=O)NC(C(=O)NCC(=O)N(CC(F)(F)F)C)C(C)C CC(CCC(C)(C)C)C(=O)NC(CCF)C(=O)N1CC2CC2C1 C(=O)(CCCCNC(c1ccccc1OC)=O)N(CCC(=O)OCC)CC c1(C(C)OC)nc(C(=O)NCC2CC(NC(C3CC3(F)Cl)=O)C2)cs1 C1(C)(NC(C(C2CCCCC2)C)=O)CC(NC(C2CCC2(C)C)=O)C1 c1(C(=O)NC(C2CCN(C(=O)C=CSC)C2)CC)cc(-c2ccccc2)[nH]n1 c1(OC)cccc(CCC(N2CC(CNC(=O)CN3CC=CC3)C3CC23)=O)c1 C1(C(N(C2CCN(C(c3ccc(C)c(O)n3)=O)C2)CC)=O)CCCCNC1=O Cc1ccc(NC(N2CCOC(c3ccc(F)cc3)C2)=O)c2[nH]ncc12 C=CC(C)N=c1cc(C)nc(NC2CC3CCC2N(C)C3)[nH]1 c1(SC)ncc(C)c(N2CC3C(C2)N3C(c2cc(O)ccc2Br)=O)n1 c1(C(=O)NCCN(c2ccnc(C(C)(C)C)n2)CCOC)ccc(OC)cc1 c1(CO)ccc(Cl)cc1CN1CCN(CC(OC(c2cccs2)=O)OCO)CC1 C1(NC(COCCC(C)C)=O)CN(C(C2C3CC(=O)CC23)=O)C(C)(C)C1 c1(C(=O)NC(CC(C)NC(c2cccc(CC)n2)=O)C)ccc(OC)cc1F Cc1sc(C)c(C(=O)NCC(C)(C(C)C)NC(c2ccc(C#N)cc2)=O)c1C N1(C(C23CC(C(N4CCC(C(=O)NC)C4C)=O)(C2)C3)=O)CCC(C)(C2CC2)C1 N1(C(c2c(C)nccn2)=O)C2CCC1CC(CNC(C1(C)C=CCCC1)=O)C2 c1(C(=O)NCC2C(C(=O)NC3(C)CC(F)C3)CC2)ccc(COC)cc1 n1(CCNC(=O)C=Cc2cccc(Cl)c2)c(CCCCl)nnc1N(C)OCC(=O)OC CCC(CC)(CCNC(=O)C(F)C1CCCC1)NC(=O)CCC#N C1(C)(NC(C(CC=C)CNC(c2ccccc2CC#N)=O)=O)CCC(=O)NC1=O c1(C(=O)NCC(CNC(Cc2nc(C)c(C)o2)=O)(C)O)ccc2occ(C)c2c1 n1(CCCC)cc(C(N2CC(CNC(c3ccn(C)c3)=O)C(O)C2)=O)c(C)n1 n1(OC)nnc2c1C(C(=O)NC1(C)CC1)CN(C(=O)CN1CCNC1=O)C2 C(=O)(C1=CC2C=CC1C2)NCC1C(C(=O)NC(CC#C)(C)C)OCC1 CCCCCCC(=O)NCCCC(O)C(=O)NC1CN(C)CC(O)C1 Cc1cccc(C)c1C(=O)NC1CCCCN(C(C2CC3CCC(C2)O3)=O)C1 c1(CC)ccc(C)c(NC(=O)CC2CC2CNC(=O)CNC2CCC(C)C2)c1 CC1=C(C(=O)NC2CCCC2NC(c2cc(C)sn2)=O)C(C)(C)CCC1 N1(C(C2C(CCN(C(=O)CCN(C3CCC3)C)C3CC3)C2)=O)CCCC1CN.CO c1(C(=O)NCC(N(C)C(c2ccnc(F)c2)=O)C2CC2)c[nH]cc(Cl)c1=O C1(CNC(CCn2ncc(C)c2)=O)CN(C(C2(NC(C)C)CC2)=O)CCN1C C1(CNC(C(c2ccn(C)n2)C)=O)CC(NC(=O)CSC(C)(C)C)CCO1 c1(NC(C2CN(C(C3CCCC4CC34)=O)C2)=O)cccc(-c2ncon2)c1 C1(C(=O)NC(C)(CNC(c2c(F)cccc2Cl)=O)C2CC2)CC(C2CCCC2)C1 N1(C(CCc2ccc(CC)cc2)=O)CCCC2(CC2NC(=O)C=C(C)C)C1 CCC(C)(C(=O)NC1C2CC(O)C1N(C(c1ccncc1NC)=O)C2)C(N)=O C#Cc1cc(C(=O)NC2CC(CNC(C3CC3c3ccc(F)cc3)=O)C2)cc(N)c1 C1(CNC(CC(=O)NCC#C)=O)CN(C(=O)C(c2ccc(Cl)cc2)CO)CCO1 Cc1cscc1C(=O)NCC(C)(CO)NC(=O)Cn1nnc(C2CC2)n1 c1(OC)ccccc1CN1CC(NC(C)CN2CCCC2=O)C1 Cc1cc(C(=O)NC2CN(C(=O)CNC(N)=O)CC2C)nn1C1CCOCC1 S(=O)(=O)(CC(=O)N(CCCN(C)C)CCNC(=O)C(C)n1cccn1)NC C#CC1(O)CCN(C(=O)C(C2(O)CCC2)NC(=O)C=CC=CC)C1 c1(CC)nc(Cl)[nH]c(=NCCC2CCCCN2C(c2ccc(C)cc2)=O)c1Cl C=CCN=C(NC(c1ccc(OC)c(OC)c1)CC(=O)OC)N1CCCC(C)C1 C1(C(N2CC(CNC(COCCCCC)=O)C(C)(C)C2)=O)CC2(COCCO2)C1 N1(C(C(C)(C)SC)=O)CCC2CCN(C(C3(C)CC4CCC(C3)S4)=O)CC2C1 N1(C(Cn2ncc(C(C)=O)c2)=O)CCN(C(c2cnc3sccn23)=O)CCC1C C(N=c1nc2c(ncn2C(C)C)c(N2CC(F)C(F)C2)[nH]1)c1c(CC)con1 Cn1ccc(=O)c(C(N2CCC2CC(=O)NC2CC(OC3CCC3)C2)=O)c1 CCCCCCCCN(C(=O)CN(C(=O)CNC(=O)C(Cl)Cl)C(C)C)C N1(C(COCCC)=O)CCCC(NC(C2C(C)C2C)=O)C1C C1(C(=O)NCc2c(C(=O)NC(c3ccoc3)C)con2)CC2CCC(C1)C2 C1(NC(C=CSC)=O)CC1C1CCN(C(C2CC(c3cnn(C)c3)=NO2)=O)CC1 CCC(O)C(C)(C)C(=O)NC(C)(C)CN1CCN(C(=O)CC23CCCC2C3)CC1 C#CCC(CC(F)F)C(=O)N1CC2CC1CN2C(c1c[nH]nc1OC)=O N1(CC(=O)NC2CN(C(=O)C=C3CC3)CC3(CC3)C2)CCc2ccccc2C1=O Cc1onc(C(N2CC(CNC(c3cc(Cl)ncc3O)=O)C2)=O)c1[N+](=O)[O-] c1(NC(C(=O)NCCC2(N3CCCCO3)COC2)=O)cncc(F)c1 Nc1ccc(C(=O)NC2(CO)CCCCC2)c(F)c1.c1(C=O)cn(CCCF)nn1 c1(OC)ccc(F)cc1C(N1CC(NC(C2CCS(=O)(=O)N2)=O)C2(CC2)C1)=O C1(OC)COCCC1NC(=O)C(C)(C)CN(C)C(c1csc(C)n1)=O C1(C(=O)NC2CC(NCCC(C)F)C23CCC3)C2C3CC4C5CC(C1C35)C24 N1(CC(=O)NCCCN(C(C(=O)NC(C)C)=O)CCO)CCCCC(O)C1=O C1(SCC)COCCC1NC(=O)C(=O)NCc1ccnc(OC2CCCCC2)c1 N1(C(CCC#C)=O)CCC(C(C2CC2)NC(c2ccc(-c3ccco3)o2)=O)CC1 N1(CC2C(=O)OCC2)CC(c2ccccc2)CCC1CO C(=O)(CCCCCc1ccccc1)N1CCCC(NC(C(C)O)=O)C1 C(N=c1[nH]cncc(OC)c1=O)c1ccc(OCC)cc1 C#CC1(C(=O)NC2CCCC2N(C(=O)CS)C)CCC1.C(C(C)(C)C)N(CC=C)CC c1(C(=O)NCC)cc(-c2ncccc2C(=O)NC(C)COC)cc(F)c1 C1(NC(c2cccnc2)=O)CN(Cc2cccc(Br)c2)C2(CCOCC2)C1 C1(CCCNC(=O)CC2CS(=O)(=O)C2)CCN(C(=O)CCOC2CCOC2)CC1 n1(C(C)C)cnc2c(C(F)(F)F)nc(NC3CCC4(CCCC4)C3)nc12 C1(C(N2CC(C=C)(O)C2)=O)CN(C(=O)CC2CCCOC2)CC12CCC2 Nc1cc(F)c(C(N2CCCC2(C)CNC(C2CCCCNC2=O)=O)=O)cc1N C12(C(N3CC(n4cc(CCCC(C)O)nn4)C3)=O)CCC(N(C)C)(CC1)CC2 C(=O)(C1COc2ccccc21)NC(CC=C)CNC(C1CCC(C)CC1)=O C=C(C)CC(C)C(=O)N1CCCCC(CNC(=O)CC(C)(C2CCC2)N(C)C)C1 N1(C(c2n(C)ncc2)C(=O)NCc2ccccc2Br)CCSCC1(C)C c1(NC)cnc(C(N2CCOCC2CNC(c2ncsc2Br)=O)=O)cn1 c1(CC2(C(N(C3CCN(C(c4ccccc4)=O)C3)C)=O)CC2)ccccc1 Cc1cc(C(c2nnnn2C)NCCCC(C)(C)OC)c(C)s1.C1(C)CCCC1 Cc1cccc(C)c1C(=O)NC1CCN(C(c2nccn2C)=O)CC1C c1(NC(C2(CC)CN(C(=O)CC(C)(C)OC)C2)=O)ccncc1C(F)F C(C(O)C(=O)N1CC=CC1CNC(=O)CC1CC1)OC C1(C(N(CC(CC)C)C)=O)CCCN1NC(=O)CC1(C#N)CC1 C1(NS(=O)(=O)Cc2cncc(Br)c2)COC2CCCCC12 CCC(F)(F)C(=O)NCCC(C(=O)N1CCOC(C(C)(C)C)C1)OC C1(N(C(=O)C#CC(=O)N(C)C)C)CC2CCC(C1)N2C(=O)CCC(F)(F)F N1(C(c2ccc(OC)o2)=O)CC2(NC(c3cccc(CO)n3)=O)CC1C2 C1(C(=O)NC(C(C)NC(c2nc(Cl)cs2)=O)CO)CCCN(CC(F)F)C1 c1(NC(=O)NCc2c[nH]nc2C(F)(F)F)cccc2nc(-c3cccnc3)[nH]c12 C(=O)(C1=CCCN(C(c2ccc(Cl)s2)=O)C1)N1CCC(O)(C(N)=O)C1 N1(C(C(c2cccc(F)c2)C)=O)CCC(C)(C)C(CNC(=O)C(C)N(C)C)C1 C12(C(=O)NCCN(C(c3c(C=C)cnn3C)=O)C3CC3)CCC(=O)N1CCS2 N1(C(C(C)NC(c2ccccc2)=O)=O)CCC(C2CCN(C(=O)C=C(Cl)Cl)C2)C1 c1(C(=O)NC(C(C)NC(=O)C2=NNC(=O)CC2)C)ccc2c(c1)CCCCN2 c1(NC(C2CC(NC(c3ccco3)=O)C2)=O)nnc(C2CCC2)s1 c1(C(=O)NCC(CC=C)NC(c2cccc(OC)c2)=O)cc(C)n(C(C)C)c1 C(C)(CCC(=O)N1CCCCC1C1CCCN(C(=O)CCn2cccn2)C1)SC C1(C(N2CCC(SCC)(CO)C2)=O)(NC(=O)CCCCCOC)CCC(F)(F)CC1 N1(C(C2CC(CNC(C(CC)(C)C)=O)C2)=O)CCCC2(CCOC2)C1 c1(CNC2CCC(NC(c3cncnc3)=O)C2)cccc2cccnc12 c12coc(c1)S(=O)(=O)C1(C)CC(C)(C1)C(=O)N1CCOC(C1)CNC2=O CN1CCC(C2(C(N3CCC(C)(NC(=O)Cc4cncn4C)C3)=O)CC2)CC1 C(CCC(C)(C)C(=O)NCC(C)C(=O)N(CC(C)C(C)C)C)OC C1(CC(=O)Nc2ccsn2)(CN(C(C)C)C(c2coc(CO)c2)=O)CCCCC1 c1(OC)cnc2[nH]c(C(=O)NCC3CCN(C(C45CC(OC)C4C5)=O)C3)cc2c1 CCC(C)(C(=O)NCCC1CCN(C(c2cn(C(C)(C)C)cn2)=O)C1)C(F)F O=C1CC(CC(=O)NC2CC(O)CN(C(c3cccc(C4CCC4)c3)=O)C2)=NN1 N1(C(C=CCCC)=O)CC(C(=O)Nc2cccc(N(C)C)c2)C(C)(C)C1 N#Cc1cnc(N2C(CNC(C3CC3C(N)=O)=O)CC3COCC23)c2sccc12 c1(OC)cc(F)c(F)cc1-n1nc(CCOC(C)C)nc1Cc1nncn1C c1(CCNC(=O)NCc2cnn(CC3CCOC3)c2)c[nH]c2c(Br)cccc12 N1(C(C2C(C(C)C)CCO2)=O)CCCC(F)(C(=O)NCC2CC23CCOCC3)C1 Cc1c(C(=O)NCCC2CCCN(C(=O)CNC(c3ccco3)=O)C2)ccn1C Cc1cncc(CC(N2CC(O)CC2CNC(=O)CCC2OCCO2)=O)c1 Cc1cc(NC(C2(C)CCN(Cc3c(Cl)ccnc3Cl)C2)=O)cc(O)c1 c1(C(N2CCCC(NC(c3c(F)cc(F)cc3F)=O)C2)=O)scc2c1OCCO2 c1(C(N2CCC(C)C2CNC(C2(O)CC2)=O)=O)ccc2nccnc2n1 c1(CC)cc(C(=O)NC2CCN(C(c3cn4c(n3)CCC4)=O)C(C)C2)ccc1F N1(C(C=C(C)c2ccco2)=O)CCC2(CCC(NC(=O)CO)CC2)CC1 C(=O)(CCS(=O)(=O)C1CCCC1)N1CC(C)C(CNC(=O)CC2CCCO2)C1 c1(OC)nc(C)ncc1C(N1CCCC(C)C1CNC(C1(C(C)C)COC1)=O)=O CONC(=O)C1=NOC(CC2CCCC2)C1.C(C)(C)(C)OC(N1CCC1)=O N1(C(c2cccc(SCCC)c2)=O)CC(NC(=O)C=CC(C)C)CC(C)C1 C1(OC)CC2CC(C1)N(C(=O)C(CCOCCO)NC(=O)CCn1cc(C)cn1)C2 C=CC1(C(=O)NCC(O)CNC(c2nn(CC)cc2Cl)=O)CCCCC1 O(NC(=O)C(CO)NC(c1ccco1)=O)CC(=C)C C1(CNC(CN(C(=O)C(C)CN(C)C)C(C)C)=O)COCC1O CC1(CNC(=O)C(F)F)CN(C(=O)CCCCc2ccccc2Br)CCO1 C(=O)(C#CC1(C)CCCO1)N1CCN(C(CCc2ccc(C)o2)=O)CC1C C1(C(=O)NCc2c(C(N(CC(CC)SC)C)=O)[nH]cc2)CC(=O)N(CC)C1 c1(OC)ccc2cc(NS(=O)(=O)C=Cc3ccccc3)ccc2c1 c1(C(N)=O)n[nH]c2c1CN(Oc1ccc(NCC(=O)O)c(OC(F)F)c1)C2 N#CC1(C(N2CC3(CCN3C(=O)CCc3nc(O)n[nH]3)C2)=O)CC12CCC2 c1(OC)ccc(C=CC(=O)NC(CO)C(C)NC(c2ccon2)=O)cc1F N1(C(C(CC=CC)CC)=O)CCC(C2CCN(C(=O)Cc3cncnn3)CC2)C1 Cc1c(NCC(N2CC(F)(C(F)(F)F)C2)=O)ncn1C C1(CC(=O)NCCCNC(=O)CCc2nc(CC3CCCC3)no2)CC2CC2C1 Cc1cc(C(=O)NCC2CCCCC2NC(c2ccnnc2C)=O)cnc1O c1(C(N2CCC(N(C(C(CC)n3cccn3)=O)CC)C2)=O)ccc(Cl)c(O)c1 Cc1cnn(C)c1C(=O)NCC1C2CN(C(C3CC3c3cccs3)=O)CC12 N1(C(CCC(C)=O)=O)CC2CCC1C(CNC(c1ccoc1C)=O)C2 c1(C(=O)NCC2CC(OC)CN2C(c2cc(O)ncn2)=O)cc(F)cc(F)c1O c1(C(=O)NC2CCN(C(=O)C(F)OC(F)(F)F)C2)cc(C2CC2)n(C(F)F)n1 C12(C(N3CCC(O)(C(C)C)C3)=O)CC(C)(CN1C(C1CCCC(O)C1)=O)C2 C12(C(N3CCCC(CN(C(=O)C(F)C4CCCC4)C)C3)=O)CCCN(CC1)C2 CC#CC1CCN(C(C2C=CCN2C(c2ccc(OC)s2)=O)=O)C1 Cc1cc(C(=O)NC(C)CCN(C)C(c2ccnn2C)=O)c(C)cc1Cl Cc1c(NCC(F)(F)Cl)nc[nH]c1=NCC1COCC1C(F)(F)F N1(C(C(C)Cc2cnc[nH]2)=O)CCCC(N(C)C(C2(C)CCC2)=O)C1 N1(C(c2c(CC)n(C)cc2)=O)CC(NC(c2ccc(CO)c(F)c2)=O)C(C)(C)C1 Cc1ccc(F)c(C(=O)NC(C)(C)CCC(=O)NCC2CCN2C(C)(C)C)c1 C12(NC(=O)CCC3CCCC(O)C3)CCC(CC1)N(C(=O)C(F)C(F)(F)F)C2 N1(CC)CCN(CC(N2CCCC(N(C)C(C3(C4CCCO4)CC3)=O)C2)=O)CC1 c1(CNC(=O)NC2CCC(C)C2)ccc(Cl)nc1 C1(C(N(C(C)C(F)F)C)=O)CN(C(C2CC(C)CO2)=O)CC1C Cc1cn2c(n1)C(CNC(C1(C)CCN(C(=O)C(=O)N3CCCC3)C1)=O)CCC2 N1(C(c2c[nH]nc2-c2ccc(Cl)cn2)=O)CCCC(C2CC2(F)F)C1 c1(OCCOC)cc(C)ccc1CN=C(NC1CCC1)NC(C1CCC1)C c1(NC(c2ccn(C)n2)C)ncccc1S(=O)(=O)N1CCC(C)(CO)C1 C1(O)(C(=O)NC(C(=O)NCCOCCOC)Cc2cn[nH]c2)CCSCC1 C1(=CC(=O)NC(C2CCN(C(=O)Cc3ccno3)C2)C)CCOCC1 c1(C(=O)NCC2(C(N)=O)CN(C(C3CCC(C)C3)=O)C2)cc(O)nc(O)n1 C1(C(N(CCC(C)NC(c2cnc3nccn3c2)=O)C)=O)Cc2ccccc2O1 C1(C(N(C(C)COC)CC=C)=O)CCCC1CNC(=O)C(C1(O)CCCC1)F c1(C(N2CC3CN(C(C4N(CC)CC4)=O)C3C2)=O)c(C)[nH]c2ccccc12 N1(C(C(C(=C)C)(C)C)=O)C2CCC1CN(C(=O)C1CCSc3sccc31)CC2 c1(OC)cc(C)cnc1C(=O)NC(C)(C)CCCNC(C1CC1(C)C(C)C)=O Cc1cc(C(=O)NC2CCCCC2NC(=O)CCC2CC2(C)C)nnc1C c1(C(N2C3CC(NC(C4CC45CCOCC5)=O)(C3)C2)=O)cccc(C#CCO)c1 c1(C(N2CCC(NC(C3(COC)CC3(F)F)=O)CC2)=O)cc(Br)cc(I)c1F C(=O)(C(C)(CSC)NC(=O)C(CC)NC(=O)OC(C)(C)C)N(C(C#C)C)C c1(C(=O)NCCOCCCNC(C(COC)COC)=O)cc(C)c(Cl)cc1F c1(C(N2C3C(NC(CC=C(C)C)=O)C(C3)C2)=O)cc2c(F)c(F)ccc2s1 C1(C)(C(=O)NCCC(C)N(C(=O)C(=O)Nc2ccccc2)C)C=CCCC1 c1(C(=O)NC2C(CNC(c3c[nH]nc3C(F)(F)F)=O)C2)cccc2cnsc12 N1(Cc2cnc(C)[nH]2)CCN(C(=O)OC(C)(C)C)C(Oc2ccccc2C)C1 C12(NC(c3c(C)nc(CCC)s3)=O)CCC(NC(c3cnco3)=O)(CC1)C2 N1(C(C(C(C)C)SCC)=O)CC(NC(C2CC=CCC2C)=O)CC2(CCC2)C1 c1(CC)cc(C(=O)NC23CC(CNC(C4CC5CCC(C4)C5)=O)(C2)C3)ccc1O C1(C(=O)NCC2(NC(c3c(C)cc(C(F)(F)F)s3)=O)CC2)CCC2(CC1)CC2 C(C(C(=O)N1CCCC(CO)CC1)C(C)C)NC(C1(CC)CCCCC1)=O c1(NC(C2C=CCN2Cc2sccc2Cl)=O)ccc([N+](=O)[O-])c2ccccc12 c1(SC)ccc(S(=O)(=O)NCCC(C)N2CCCC2)c(Cl)c1 C1(C(N(CCN(C(=O)C(O)CN2CCOCC2)CC)CC)=O)CCCC(CF)C1 N1(C(C(C)=C(CC)C)=O)CC(C(=O)NCC2(C(C)C)CC2)C(F)(F)C1 N1(C(C(c2cccnc2)NC(C2C(CCC)C2)=O)=O)CCCc2occc2C1 N1(C(c2c(C)n(C3CC3)nc2)=O)CCC(NC(=O)CC2=CCCC2)C(C)C1 CC1CCC(CNC(c2cc(N)ccc2F)=O)N(C(c2cc(Cl)cnn2)=O)C1 N1(C(c2scc(C)c2C)=O)CCC2C(NC(c3ccnc4[nH]cnc34)=O)C2CC1 C(N=c1[nH]c(=NC2CC3(CCOC3)C2)c2ccccc2[nH]1)C1(OCCOC)CC1 C(CN=[N+]=[N-])(C(=O)NCC(N1CCCC1)C)NC(CCCOCCOC)=O c1(NCC(C2CC(F)(F)C2)OC)nccc(=NCCC2CCCC2O)[nH]1 C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(c2cnc(C)nc2O)=O)CC12CC2 C(=O)(C(COC)(CC)CC)N(CC(CN(C(c1cnc(CC)nc1C)=O)C)O)C Cn1c(CN2CCN(Cc3nc4ccccc4s3)CC2)nc2cccc(Cl)c12 N1(C(CCCS(N)(=O)=O)=O)CCC2(CC1)OCCC2NC(c1occc1Cl)=O C(=O)(C1=NOC2(CCOC2)C1)N1C2C(NC(=O)Cc3c(F)cccc3F)C(C2)C1 C1(NC(c2n(C)nc(C(F)(F)F)c2)=O)COC2(C1)CN(C(C1(F)CCOC1)=O)C2 C12(CNC(c3n[nH]cc3[N+](=O)[O-])=O)CCC(CN(C(=O)C3=COCCO3)C1)C2 C(C(C)(CNC(C1(CNC(=O)C(=O)C2CCCC2)CCCC1)=O)CO)OC c1(C(=O)NCCCC(C)NC(c2ccc(Cl)cc2)=O)cc(Cl)cc(Br)c1 C1(CC#N)COCCN1CC(=O)NC1(O)CCN(S(=O)(=O)CCCCl)C1 c1(COCC2CC(F)(F)C2)ccc(S(=O)(=O)NCC(C)C(F)F)cc1F N1(C(c2cn(CCC)nc2)=O)CC2CC1CN2C(=O)C(c1ccc(C)cc1)C n1(C(C)C)cccc(NC(c2nnnn2C2CC2)CC2CCC(F)(F)CC2)c1=O C12(C(=O)NC3CC(CNC(CCC=C(C)C)=O)CC3O)CC3CC(CC(C3)C1)C2 Cc1ccc2ccccc2c1CC1CC1C.N12CC3C(C3C1)C(C(=O)O)C2=O Cc1ccc(C)c(OCC(N2CCN(C(C3CCCS3)=O)C(C(N)=O)C2)=O)c1 CC1CCc2nc(C(=O)NC3CN(C(c4cnco4)=O)C(C)(C)C3)cn2C1 c1(C(N2CC(C(N)=O)(CNC(C3CCC(C)C3)=O)C2)=O)cccc(CO)c1 CC(C)S(=O)(=O)CC(=O)N1CC2(CCN(C(=O)CC(c3ccccc3F)C)C2)C1 c1(C(CN(C(C(C2CC2)OC)=O)C)O)ccc(C)cc1 C1(C2CC2)(CNC(C(COC)(C)C)=O)CCN(C(c2c(C)cccc2C)=O)C1 O=C(C1CSc2ccccc21)N1CCN(C(C2CC3COCC(C2)C3)=O)CC1 CCC(C)C(C(=O)N1CCCC(C)CC1)OC Cc1nn(CC(=O)NCc2cc(C(=O)NCC3(C)CC3(C)C)on2)c(=O)o1 c1(C(N2CCC(O)(C(C)NC(C(CC)N(C)C)=O)C2)=O)cc(O)c2ccoc2c1 c1(CN(C(C2C(OC)C2)=O)C)ccc(CNC(c2cn(C(C)C)cc2C)=O)cc1 S(=O)(=O)(c1ccc(C)cc1)NCCC(N1C2CN(C(C=CCOC)=O)C(C2)C1)=O C(=O)(C(CO)C(F)(F)F)NCCC1(C)CCN(C(C2OCC(C)(C)C2)=O)C1 c1(OC)cc(N(Cc2cc[nH]n2)Cc2nncs2)cc(F)c1 c1(C(=O)NCC2C(NC(c3nccc(N)c3)=O)CCC2)cc2cnc(Cl)cc2s1 N1(C(C(C(C)C)NC(N)=O)=O)CCCCC(CNC(=O)COCC(F)F)C1 C=C(C)CCCC(=O)N1CCOCC1CNC(=O)CCCn1ccnc1C c1(C(=O)NCc2nnc(COC)s2)c(Br)nc(C)n1C N1(C(CN(C2CCCC2O)C)=O)CCOCC1CNC(c1cc(Br)n(C)c1)=O C(=O)(CCN(C(=O)CCn1cccn1)C)N(CCOC)CCC(F)F c1(OC)ncccc1NC(C1CC(C)N1C(=O)Cc1sccc1C)=O CCCC(F)C(=O)N1CCSCC1C(=O)NC1CC2CC1CO2 N1(C(c2cc(C)cc(Br)n2)=O)CC(C)Cc2cccc(O)c21 C(CC1CCOCC1)(C(=O)NCC1CCCO1)NC(C1(COC)CC1)=O N1(C(CONC(=O)CCCSN2CCCC2=O)=O)CCC(C2CC2)C1 C[S+](C)CCC(O)C(=O)N1CCCC(NC(C2CCN(C(N)=O)CC2)=O)CCC1 C1(CC(N2CC(c3cn(CCCCC(=O)O)nn3)(O)C2)=O)CC2(C1)CC(CO)C2 c1(C(N2CCC(NC(C)=O)C(F)C2)=O)cc(F)c(F)cc1Cl.c1cc(Cl)cn1C C1(CC(=O)NC(C2(O)CN(C(C3(NC(N)=O)CC3)=O)C2)C)CC(C)(C)OC1=O N1(C(C2(F)CCN(C(CC3(NC(C)=O)CC3)=O)C2)=O)CC(S(C)(=O)=O)C1 n1(CCC#N)c(N2CCOC(n3cncn3)C2)nnc1-c1cccc(Br)c1 Cc1ccc(NC(=O)C(C2CC2)NC(c2ccc(C#N)cn2)=O)cc1C N1(C(C2C(OCC)C2C)=O)CCCC2(C1)CN(C(c1ccc(CC)s1)=O)C2 C(CCN=c1[nH]c2ccc(F)cc2s1)N1CCN(C(C(C(=C)C)(C)C)=O)CC1 c1(NC(=O)NCCCc2c(C)ccnc2)cnc(Cl)c(C(F)(F)F)c1 C12(C(N(C3C4CN(C(c5cn(CC)nc5)=O)CC43)C)=O)CC(C1)C(C)(C)O2 C1(NC(C=CC)=O)CCN(C(=O)CSc2cc(-c3ccccc3)oc2C)C(C)C1 C1C(C)(C)CCN=C(NC(C)C2CC2)N1.C1(OC)CCN(S(C)(=O)=O)C1 C1(N(C2CCC3(CC2)CNC3)C(C)=O)CC2CCC(C1)N2C(=O)C(Cl)Cl c1(CNC(CC(C=C)C)=O)c(C)nn2c1CN(C(=O)CCCCN(C)C)CC2 Cc1cccc(F)c1CC(N1CCC(C)(NC(=O)CCNCCCC(N)=O)C1)=O N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(C)CC1C(=O)N(CC(O)CN(C)C)C C=CCCC(C)(C)CNC(C1C=CCCN1C(=O)Cn1cnnn1)=O C(=O)(C1=NOC(C2(O)COC2)C1)NC(CN(C(c1cnc(OC)cn1)=O)CC)C c1(CC)ncncc1C(=O)NCC1CC1CNC(C1CCCCC1)=O Cc1oc([N+](=O)[O-])cc1C(=O)N(CCCNC(=O)C(O)C(C)C)CC1CCCC1 CN1CC(NC(=O)C(C(C)(C)C)NC(C23CSCC2C3)=O)C2(CC2)C1=O c1(OC)cc(NC(C2CN(C(=O)Cc3nncs3)CCO2)C)ncn1 c1(N(CC(=O)NCC(Cc2ccccc2)NC(CC=C)=O)C(C)=O)ccccc1O Cc1nsc(C(N2CC(O)(C3CCCO3)C2)=O)c1N.c1(C2CN2)n[nH]c(=N)s1 c1(C(=O)OC)cc(C(N2CCN(C3CC3)CC2)C(=O)NC(C)(C)C)ccn1 C1(OC)CCCC1C(=O)N(CCCc1cn(CCCCF)nn1)C1CC1 Cc1cc(C(N2CC3CC(NC(c4cnc5n4CCS5)=O)C2C3)=O)cn(C)c1=O c1(C(N(CCC(C)NC(C(F)=C(C)C)=O)C)=O)c(C)ccc2c1CCCN2 N1(C(CCC=CC)=O)CC(NC(c2cc(OC)n(C)n2)=O)C(CCC)C1 Cc1cncc(C(=O)NCC2CN(C(c3ccc(CO)cn3)=O)CC2O)n1 C1(C(=O)NC2C(C)CN(C(C3CN4CCC3CC4)=O)C2)Cc2nn[nH]c2C(C)C1 C(CC(=O)N1CCC(O)(CCNC(C2COC(C)(C)C2)=O)CC1)(C(F)(F)F)OC C1(NC(C2CC(CCC)C2)=O)CCSC12CN(C(=O)C(n1ccc(C)n1)C)C2 c1(C(N2CC3(CC(NC(CCC(C)SC)=O)C3)C2)=O)nccc2cccnc12 N1(C(C(CC)(C)O)=O)CCOC2(CCN(C(=O)Cc3cncc(Br)c3)C2)C1 CCCCCS(=O)(=O)CC(=O)N(C1CCCN(C(c2cc(=O)n(C)o2)=O)CC1)C c1(C(=O)NC2CC(NC(C3OCC(C)OC3)=O)C2)cc(=O)c2ccncc2o1 c1(OC)cc(C(N2CC(CCNC(c3cnc(Cl)[nH]3)=O)OC(C)C2)=O)ccc1Cl C1(C(=O)NCCN2CCOCC2)CC12CCN(C(c1cccc(I)c1)=O)C2 C1(CC)CCOC1C(=O)NC1(C)CN(C(C2CN(CC(C)C)C2)=O)C1 C#CC1CC2(CC2)CN1C(c1ccnc(C(F)F)c1)=O c1(C(=O)NCC(C)NC(=O)CC2CCC2(F)F)ccc(O)nc1 c1(CCC)nc(C(=O)NCC2(NC(C3CCC(F)C3)=O)CCCC2)co1 C(C1CCCN1C(=O)CCc1nc(O)n[nH]1)=CC(NOCCC#C)=O C=CC1(CO)CCN(C(c2[nH]nc(C(F)(F)F)c2C)C(=O)NCC2CC2)CC1 C1(n2cc(C(N)=O)nn2)CCN(C(=O)C(=O)NC2CCCCC2OC(F)F)CC1 c1(C2C(C(N3CCC(N(C(CN(CCOC)C)=O)C)C3)=O)C2)ccc(C)cc1 N1(C(CC(CC#C)NC(=O)C(C)(C)NC(C)=O)=O)CCC2(CC1)CC(O)C2 C1(CNC(c2c(C(C)C)occ2)=O)CC(C(=O)NC(CN(C)C)CCO)=NO1 N1(C(c2cc(CC)oc2C)=O)CCN(C(c2cnc(Cl)s2)=O)CC1C(F)F C(=O)(CC1=NNC(=O)C1)N1CCC(OC)(CNC(=O)C(C)c2cccs2)CC1 c1(C(=O)NCC23C(CN(C(C(=Cc4ncn(C)c4)F)=O)C2)C3)cn2c(n1)CCC2 C(CCCS(=O)(=O)CCO)NC(C1CCN(C(c2ccncc2F)=O)CC1)=O C1(CNC(=O)C(O)Cn2cncn2)CN(C(c2sc(F)cc2Cl)=O)CCO1 N1(C(C2C(=C)CC2)=O)CCC(C)(C)C1CNC(c1cc(C(C)C)nn1CC)=O CC1CC(NC(=O)CC2OCCC2C)CN1C(=O)Cn1cc(CO)nn1 CN1CC2CCN(C(=O)CCN(C(c3c[nH]c(=N)o3)=O)C3CC3)CC2C1 c1(-c2ccc(N(c3ncc(C4CCOCC4)o3)C(C)C)cc2)ccc([N+](=O)[O-])cc1 N1(C(c2cc(OC)cc(Cl)c2)=O)C2CCC1CN(C(=O)C(C)OCC(C)C)C2 c1(OC)cccc(NC(C2CCN(C(C3COC(=O)C3)=O)CC2)=O)c1F c1(C(N(C(C)CNC(c2cocn2)=O)CC)=O)ccc(N)c2ncccc12 N1(C(C(CC)CC(F)F)=O)CCN(C(c2ncoc2C(F)(F)F)=O)CC(C)(C)C1 CCC1=NOC(C(=O)NC2CC(C(F)F)(NC(=O)Cc3cnn(CC)c3)C2)C1 c1(CNC(=O)Nc2c(OC)nc(Br)cn2)cc(Cl)c(C)c(Cl)c1 CC1CCc2ccccc2N1CCN=C(NC(c1ccc(Cl)cc1)=O)NC1CC1 C1(C(N(C(c2ccccc2)CNC(Cc2c(C)non2)=O)C)=O)CC(F)C(=O)N1 C=C(C)CCCC(=O)N1CCC(C2CCCN2C(=O)CCCOc2ccccc2)C1 c1(C(=O)NC(C(C)NC(c2cn(CC=C)nc2)=O)CO)cc2ccccc2nn1 c1(C(=O)OC)ccc(CNC(=O)NN2CCC(OC(C)(C)C)C2)o1.C(Cl)=C CC1(C(N2CCC(O)C2C(=O)NCCc2cocn2)=O)CCC2CC2C1 C1(C)(CNC(C2C(CC)C2)=O)COCCN(C(c2nocc2C(C)(C)C)=O)C1 C(=O)(C(C)(O)C(C)(C)C)NCC(C(C)(C)C)NC(c1nc(C(F)(F)F)cs1)=O C1(NC(c2nc(C(C)(F)F)sc2)=O)CCCCC1NC(=O)C(F)C1CC1 CCC(C)C(C)CNC(C1COCCN1C(=O)CC(C)OC)=O c1(NC(CCCC=C)c2nnnn2Cc2ccco2)ccc2oc(O)nc2c1 C1(O)(C(C)NC(=O)Cc2csnn2)CCN(C(c2nc[nH]c2C(C)(C)C)=O)C1 c1(OC(C)C)ccc2c(c1)OCCN2C(c1coc(-c2cnn(C)c2)n1)=O C1(NC(CCN(S(C)(=O)=O)C)=O)CCCCC1NC(=O)C=CS(C)=O Cc1cc(=NC(=O)CC(C)N(C)C(c2nccn2C(C)C)=O)[nH]n1C1CC1 C1(NC(c2c(C)ccnc2)=O)CCN(C(=O)Cn2cncc2C)CCC1(F)F c1(C(N2CC(O)(C(C)(C)CNC(C3C(C)(C)C3(F)F)=O)C2)=O)ncnc(O)c1F CCC(c1cccc(Cl)c1)=CC(=O)NCCC1CC(NC(c2[nH]cnc2C)=O)C1 C(=O)(C(CC)SC)NCC(C)(C1CC1)NC(C1C(C=C)C1)=O C=CCCCC(C(=O)N1CC(OCC)C1)NC(=O)C(C1CCC1)OC(C)C c1(C(N2CCC(c3ccco3)C2)=O)ccc(C=CC(=O)NCCCC)cc1 N1(C(COCCN(C)C)=O)CC=CC(C(=O)N(C2CCC2)C2CC2)C1 Clc1c(NC2CCNC3CC23)cccc1I c1(OCC)ccc(CN(CC(C)C=C)C(=O)C(=O)NCCS(C)(=O)=O)cc1 c1(C(=O)NCC(CO)NC(C(C2CCC2)OC)=O)cc(-c2ccn(C)n2)on1 C12=NC(=NCC3(CCC3)N(C)C3CCN1CC3)Nc1cc[nH]c12.CN.SC C(=O)(C1=NOC2(CCC2)C1)NCCCCC(C)NC(c1n(CCC)ncc1)=O Cc1cc(C(=O)NCC(c2ccccc2)CNC(C23CCC2C3)=O)c(C)cn1 C1(NC(C2CCC(=C)CC2)=O)CN(C(C2CCOC(=O)N2)=O)CC2CCCC12 C(=O)(C(F)(F)c1cccnn1)C(c1c[nH]nc1N1CCNCC1)=O.N C(=O)(CCC(=O)N(C)CC1CCCN1C(=O)CC1CCNC1=O)NC CCCN=C(NCC(Cc1ccc(Cl)cc1)CO)NCC(F)CO CCCC(C)(O)CNC(=O)C(C1CCCN(C(C2(Cl)CC2(F)F)=O)C1)C C1(C(N2C(C)CC(NC(=O)C(F)(F)C3(O)CCC3)C2)=O)CC12CCCCCC2 C1(C(=O)NC2C(C=C)OCC2)CN(C)CCN1C(c1nccc(C)c1F)=O c1(C(=O)NCC23N(C(C4CCCC(C)CC4)=O)CC(C2)C3)cncc2c1CCC2 C(CCCCC(=O)NC1CN(C)CC1C)OC c1(C(=O)NC(c2cn(C)nn2)C(N2CC(OCC(=O)NC)C2)=O)cn(C)c(C)n1 c1(C(=O)NCCC(C)(C)NC(C(C)NC(COC)=O)=O)cn(CCOC)nc1C c1(NC(=O)CC2CN(C(=O)CCc3ccc(F)cc3Br)C2)cccc([N+](=O)[O-])c1 N1(C(CSCC=C)=O)CC(C2(NC(c3cc(O)cc(Cl)c3)=O)CC2)C1 C1(C2CCN(C(=O)CC3CCOCC3)CC2)(NC(C(C)=C2CC2)=O)CCC1 CC1CN(c2cc(N3CCC(c4nc(=N)[nH][nH]4)CC3)ncn2)CCC1(F)F N1(C(c2c(C)n[nH]c2)=O)C(C(=O)NCC2(CO)CCN(C)C2)CCC1C1CC1 C1(CC(C(=O)OC)O)CCN(Cc2n[nH]cc2C2CCCC(=O)N2)CC1 CCCCC(C(=O)Nc1cccc(Cl)c1)N(C)Cc1ccccc1N(C)C c1(CNS(c2ccc(CSC)s2)(=O)=O)nc2ccccc2nc1C c1(C(N2C3CC(N(C(C(C)O)=O)C)CC2CC3)=O)cn(C)c(=O)c2ccccc12 C1(n2cc(C34N(C(CC(C)C(F)F)=O)C(CC3)CC4)nn2)CC2CC1CC21CC1 c1(C(=O)NCC(CNC(COCCOC)=O)CO)nc(Cl)ccc1OCC1CC1 c1(NCc2c(C)nco2)nccc(N2CCCC(c3cc(C(F)(F)F)[nH]n3)C2)n1 N1(C(c2scc(C)n2)=O)CC2COCC2(C(=O)NCC(C)S(C)(=O)=O)C1 CC1(OCC(=O)NC2CC(CC(=O)N(C3CCOC3)C3CC3)C2)CCCC1 c1(C(=O)NCC2CC(O)(CNC(C(CC=C)CC)=O)C2)c(C)cc(C)nc1C c1(CC)ccc(C=CC(=O)NCCC(C)NC(c2ncc[nH]c2=O)=O)o1 C1(C(=O)NCc2cnc(CO)o2)CCC2CC1CO2.C12CCC(C1)NC(=O)CC2 N1(C(C(C)NC(C)=O)=O)CCN(C(=O)C(C2CC2)Sc2ccccc2)C2(CC2)C1 N1(CCCSC2CC2)CCCCCC1=O.n12cc(nn1)CN1CCC(C1)NC(=O)C2 N1(C(CC=CCC)=O)CC2CC1C2NC(C1CC1C(C)(C)C)=O C1(NC(CC(=O)NCC)=O)CCC2(CC1)CC2NC(c1ccnn(C)c1=O)=O CN=c1[nH]ccc(C(N2CC(C(N)=O)(CNC(=O)C(F)OC)C2)=O)c1N c1(C(N2C(CNC(c3cn(CC)nn3)=O)CC2)=O)ccc2c(c1)NC(=O)C(C)O2 N#Cc1cc(F)ccc1CN1CCOCC(NC(=O)C=Cc2cccc(O)c2)C1 C1(C2CN(C(C3CC(=O)N(C)C3)=O)C2)(NC(C(C2CCCCCC2)OC)=O)CC1 C1(CNC(Cn2cnc(C)n2)=O)CC2CCC1N2C(C1CN(C)C1)=O CCCC(C(=O)NCCC(O)C(=O)NCc1coc(CC)n1)OCC c1(C(=O)NC2CC(F)CN(C(=O)C=Cc3cocn3)C2)ccc2nccn2n1 N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(CO)C(NC(=O)C(N)=O)C1 C(CC(C)(C)CC(=O)N1CCN(C(c2cccc(C(F)F)c2)=O)C2CC12)OC C1(CNC(CC2(C)N(C(C3(C(C)=O)COC3)=O)CC2)=O)CCCC12CC2 C1(CNC(C2(C)CCC2)=O)CC12CCN(C(=O)Cc1nnc(O)s1)CC2 C=C(Cl)CCC(=O)NC(C)CCN(C)C(c1cc(C)n(-c2ccc(F)cc2)n1)=O Cc1cnc(C(N2CCC(C)(NC(C3CC4OC3C3CC43)=O)C2)=O)cc1C c1(CC)cccc(CNC(C2(CC)CCN(C(=O)C=CC(C)C)C2)=O)c1 C1(CNC(CC#C)=O)CN(C(=O)C(C)Cc2ccc(OC(F)(F)F)cc2)CCO1 c1(CNC(C2C(CCC)C2)=O)ccc(C(=O)NCC(C)(C)NC(C)C)nc1 N1(CC(NC(=NC)NC2CCc3ncnn3C2)=O)CC2C3C=CC(C3)C2C1 C12(NC(c3ccc(CC)[nH]3)=O)CCCN(C(C3(C)CCS(=O)(=O)CC3)=O)CC1C2 c1(C(=O)OC)nc(N(C(C)CNC(c2cnc(Cl)s2)=O)C)ncc1Cl c1(N(C)CC2CC2(F)F)cc(S(=O)(=O)NC2CCCS2)ccc1C#N C(CCCC(=O)NC1CCCCC1CNC(=O)CC1CC2(CC2)CO1)NC(N)=O C1(C(N2CC(N(C(COCCC(C)C)=O)C)C(C)CC2)=O)CN(C)C(=O)CCO1 C(=O)(CC(C)CCc1ccccc1)NCC1CN(C(Cc2cccc(C)c2)=O)C1 c1(C(N2CC(NC(CC(C=C)C)=O)C(C)(C)C2)=O)cc(C)nc2c(O)cccc12 CN1CCN(C(=O)CC2CSCCO2)C(C(=O)NCc2ccnc(F)c2F)C1 c1(C(=O)NC2CC(C)(C)N(C(c3ccc(N)cc3F)=O)C2)ccc2c(c1)OCO2 c1(C(N(CCOCCNC(C(CC)NC(N)=O)=O)C)=O)cccc(OC)n1 c1(C(N2CCC(NC(c3cc(C4CCC4)[nH]n3)=O)C2)=O)cc(C2CCOC2)[nH]n1 N1(C(c2ccc(NC3C(CC)C3)cc2)=O)CCOC2CN(C(=O)C(C)(C)F)CC12 C1(NC(CNC(=O)OC)=O)CCCC1NC(=O)COC1CCCOC1 N1(C(C)=O)c2ccccc2CC1C(=O)NCC1(NC(c2ccc(C#N)s2)=O)CC1 Cc1cccc(C)c1CNC(=O)CC1CCCC1NC(C1CCCC(O)C1)=O CC(C)(C)S(=O)(=O)CC(=O)N1C2CCC1CN(C(c1cccn3cnnc13)=O)C2 N1(C(=O)NC2N(C(C3CC(C(=O)OC)C3)=O)CC3(CC3)C2)CCN(C)C(=O)C1C c1(C(=O)NCC(=C2CN(C(C3(CC#C)CCCO3)=O)C2)F)ccccc1C N1(C(CCC(=O)NCCC)=O)CCN(C(=O)C2=NNC(=O)CC2)CC(CO)C1 c1(C(N2CCCC(CNC(CCOCC#C)=O)C2)=O)ccc2c(c1)CN(C)CC2 c1(CC)ccc(C(=O)N(C)CC2(O)CN(C(=O)C3=CC(C)C3)C2)c(Cl)c1 CCCC(CNC(c1c(C)cnnc1O)=O)C(=O)N1CC(O)CC1(C)C c1(CCC(N2C3CN(C(C4(C#C)CC4)=O)CC2CC3)=O)nc2cccc(Cl)c2[nH]1 O=C(CCCC(F)(F)F)NCC1CC2CCCC2N1C(=O)CSc1n[nH]c(O)n1 C(=O)(CC(C)(C(F)F)N(C)C)N1CCCC(O)(CN(C(CC)=O)C)C1 C1(C(=O)NC(c2nocc2C(=O)NCc2ncccn2)C)CC(=O)NC(=O)C1 C1(CC(=O)NC2CCN(C(c3c(C)scc3)=O)C2)CCNC(=O)C1 c12cc(cnc1O)NC(=O)NNC2=O.C1(CC(C)(C)C)CC(C(=O)O)CCO1 Cc1cc(C(N2CC(NC(=O)CC3CC4(CCC4)CO3)CC(C)C2)=O)cc(N)c1 Cc1csc(CCNC(=O)C(CC2CC2)NC(C2C=CCCC2)=O)n1 c1(C(=O)NCCCN(c2ncc(C#N)cc2F)CC)cccn2nnnc12 C1(NS(CC(C)c2ccc(F)cc2)(=O)=O)CCCc2ccccc2C1 Cc1nn(C)c2c(NCC3CC4C=CC3O4)nc(=NCC3C(C)C3C)[nH]c12 N1(C(C2CCN(C)C2=O)=O)CC2(CCCC2)C1C(=O)NCC1(C(N)=O)CC1 CC1(O)CC2CC1CN2C(=O)NC(c1ccccc1Cl)CO C1(NC(=O)COC)CCc2cncn2C1.c12cc(n[nH]1)C(=O)N(CC)C2 Clc1cc[nH]c1C(c1nnnn1C1CCCC1)NCC1(CCO)CCC1 C1(C(=O)NCC(C2CC2)NC(C(CC)O)=O)CCN(c2ncccn2)CC1 c1(C(C(=O)N(C)CCNC(C2(c3nccs3)CC2)=O)(F)F)cn(C)nc1C(F)(F)F C1(CNC(c2ccc(C)cc2)=O)CN(C(C2CC2C#N)=O)CC2(CCC2)O1 C1(C(=O)NC(CC(C)C)CO)C2CCCC2CN1C(=O)CCC1CCCC1 N1(C(c2c(C#N)ccs2)=O)CCC(CO)(NC(c2cc3[nH]ccc3s2)=O)CC1 C1(CNC(CCn2c(C)ncc2)=O)CN(C(=O)C(F)C(F)(F)F)CC(C)(C)C1 C(CC(C)(C)CC(=O)N1CCC(C(N2CCC(NC(C)=O)CC2)=O)CC1)OC n1(CC)nnc2c1CCC(C(=O)N(CCCNC(=O)CC1CCC1)C(C)C)C2 C(=O)(C1CCc2nc(C)[nH]c21)NCC1C(NC(CCCOCC)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)NCCCC(C)NC(c1ccc(C)c(C)c1Cl)=O C1(NC(c2cn(CC=C)nn2)=O)CCCC12CN(C(c1ccc(C)c(N)c1)=O)C2 C1(CC(=O)NCc2nccc(C(=O)NC3C4CCCC34)c2)Cc2nccn2C1 c1(C(N(C)CC2CCN(C(c3ccc(C(N)=O)o3)=O)CC2)=O)cc2n(c1)CCC2 N1(C(C2(C)CCCO2)C(=O)NCCC)CCC12CCC(O)CC2 CC(C)CC(C(=O)NCC1=CCCN(C)C1)ONC(C1CCCOC1)=O C(=O)(C(C1CN(C(=O)C=CCOC)C1)OC)N(CC#C)CCO.C1(OC)(CO)CCC1 N1(C(c2nc(CC)sc2)C(=O)NC2(C)CC2)CCOC2CCN(C)CC12 N1(C(C(C)(C)C2CC2)=O)CCCC(F)(CNC(C2CS(=O)(=O)CCO2)=O)C1 CN1CCC(C(N2CC3C(C(N)=O)C3C2)=O)(NC(=O)CC2(C)CCOCC2)C1 c1(CC)cc(=O)oc2cc(CC)ccc12.c12cc(Cl)c(cc1Cl)oc2=O C1(F)(C(=O)NCC2C(CC(=O)NCc3ncn(CC)n3)C2)CC=CCC1 CN1CCCC(C(=O)NCC2(O)CN(C(C3(C(F)F)CCCO3)=O)C2)C1 C1(C(N2CCCC(C3N(C(C(CC)(C)C)=O)CCC3)C2)=O)Cc2cccnc2C1 c1(OC(C)C)ccc(C(=O)NC2CN(C(=O)Cc3cccn3C)CC2O)cn1 CCCCC(C)C(=O)NC1CCOC1C(=O)NC1CC12CCCC2 C(C(=O)NCCC1(CNC(=O)C=CS(C)=O)CC1)(C(C)(C)C)N1CCC(C)CC1 C(=O)(CCC(=O)N1CCOCC1CCNC(c1ccc(C(C)N)cc1)=O)NCC c1(C(N2CC(NC(C(CCC)C)=O)C(F)CC2)=O)cc2c(cc1N)CCC2 C(=O)(CC1OCc2ccccc21)NCCCOCCN(c1ncc2[nH]ncc2n1)C N1(C(CN(C(C(C)C)=O)C)=O)CCC2(CO)CN(C(c3scnc3Cl)=O)CC2C1 Cc1cnnc(C(=O)N(C)CC2CC(F)CN2C(c2cn(C)nc2C)=O)c1 C1(NC(c2c(CNC(C3C(C)OCCO3)=O)noc2)=O)(CO)CCCCC1C N1(C(Cc2cccc(C#C)c2)=O)CCN(C(=O)C2=CCCCO2)C(C)C1C C1(C(=O)NC(CC)(C)CNC(=O)CC2=CCCC2)CCC(=O)N(C)C1 c1(C(=O)NCC2C(NC(CCOCCOC)=O)CC2)ccc(S(N)(=O)=O)cc1 CCC(CC)C(C)C(=O)N(C)CCNC(=O)Cn1cc(CO)nn1 c1(CC(=O)NC2CC(NC(c3c(C(C)=O)cncc3)=O)C2)ccccc1S(C)=O C1(NC(CC2(NC(=O)CCCc3ccc(F)cc3)CCC2)=O)CCC(=O)NC1=O c1(C(N2CCN(CC)CC2)C(=O)Nc2ccc(C#N)cc2)cccc(C)c1F CC1CC2CN(C(C3CC4CCC3C4)=O)CC2N1C(=O)C1Cc2ccccc21 N1(C(CCNC(C)=O)=O)CC2CCC1C(CNC(=O)C(C)SC(F)(F)F)C2 CC1(C#N)CCN(C(C2CC3CC3N2Cc2ccc(O)nc2)=O)CC1 C1(NC(C(C=C)C)=O)CN(C(=O)CCCN(C)C)C2CC12 C#CCCCC(=O)N1CC(O)(CCNC(c2cc(C)co2)=O)C1 C1(N(c2cccc(CO)c2)C(c2ccc3[nH]ccc3n2)=O)COC2(CCNCC2)C1 C=C1CCC(C(=O)NCCC2CC(C(=O)N(C)CC3(O)CCOC3)C2)CC1 C(C(CC(C)C)C(=O)N(CC(=O)NC1CC1)C)NC(c1c(C#C)c[nH]n1)=O C12(NC(C3CCCC(OC)C3)=O)CCCCC1N(C(=O)OC(C)(C)C)CC2 C1(C(=O)NCCCNC(=O)Cc2cn3c(n2)CCCC3)CC12CCS(=O)(=O)CC2 CN1CC(C)(C(N2CC(NC(=O)CSc3ccc(Cl)s3)C2)=O)CCC1=O C(=O)(CCCCC(F)(F)F)NC1CN(C(C23OC(C)C(C2)C3)=O)CC1C c1(CC)cccc(CC)c1CC(=O)OCC1CC1CCCCC(=O)OC N1(C(C=CC)=O)CCCC2(C1)CN(C(C13CCS(=O)(=O)CC1CNC3)=O)C2 C1(CC)C(C(=O)NC(C)C(C)F)CCN1C(=O)Cc1cscn1 Cc1nccc(Cl)c1C(=O)NCCC(C)NC(c1ccnc(Cl)c1N)=O N1(Cc2cc(OC)ncn2)CCC2CN(C(=O)CCc3cccc(C)c3)CC2C1 c1(CCC)cccc(C(=O)N(CC(C)CNC(c2cnc(C)s2)=O)C)c1 c1(C(N2CCCC(NC(C(C)C3CC3)=O)C2C)=O)cc2cc(N)ccc2o1 c1(C(=O)NCCC(CC)(C)NC(=O)C2=C(Cl)CCC2)ncc(Cl)cc1F c1(N2C3CN(C(c4cnc(C)[nH]4)=O)C(CC3)C2)ncnc2cccnc12 N1(C(c2ccc(C)c(C)c2)=O)CC2CCC(C(=O)NCCCc3nncs3)(C2)C1 C1(C(=O)NCC(CCCC)NC(c2ncsc2C(C)C)=O)CC2CCCC(C1)C2 CC(CC=Cc1ccccc1)C(=O)N(C1CCCN(C(c2ccccc2)=O)C1)C n1(CC(N2CC=CC(C(=O)Nc3cccc(OC)c3)C2)=O)cnc2ccccc12 c1(C(=O)NC(CC)CNC(C2(COC)CCCO2)=O)nc(C)ccc1F C(=O)(C(CO)C(F)(F)F)NCCC1(O)CCN(C(c2c(C)n(C)nc2)=O)CC1 C1(C(=O)NCCCCC(C)NC(C23CC(C)(C2)C3)=O)CCCC(F)(F)CC1 c1(OC)cccc(N(C(=O)C=C(C)CNC(C2CCC(C)(C)C2)=O)C)c1 c1(C(=O)NC(C(C)NC(CC2CC(=C)C2)=O)C)c(OC)ccnc1F C1(CNC(C2C(CC)C2)=O)CC(C)CN1C(=O)CC(F)(F)Br N1(C(CCCc2n(C)cnn2)=O)CCC(O)(CCNC(c2csc(Cl)c2)=O)C1 C1(C(=O)NCC2N(C(c3c(C)n(C)nn3)=O)CCC2C)CCC(=O)C(C)C1 CCC(F)(F)C(C)(C)C(=O)Nc1cnn(CC(C)(C)C(F)(F)F)c1.c1(C2CNC2)ccncc1 c1(-c2cn(C(C(=O)N(C)Cc3ccc(Br)s3)C)nn2)ccn(C(=O)OC(C)(C)C)n1 c1ccc(CNCC2CCCN2Cc2cccs2)cc1 N1(C(c2c(OC)c(O)nc(O)n2)=O)CCC2(CC1)COC(C)C2 C#CCCCCCC(=O)N1CCCC1C(C)(C)NC(C1CCc2nn[nH]c2C1)=O CCC(C)CC(C)N(C(c1ccccc1OC)C(=O)N(CC)CC)C c1(CC)ccc(C(N2CCC(CN(C)C(C3(C)CCCS3)=O)CC2)=O)cc1CC CC(C)S(=O)(=O)C(C)C(=O)N1CCN(C2CN(C(=O)CCc3ccsc3)C2)CC1 CON(C(=O)C1=NOC2(CCN(C(=O)OC)C2)C1)C=O.C(C)(C)(C)C=O c1(NCC2(C(=O)OC)CC2)ncnc2c1ncn2CC(O)C(C)(C)CO CCCC(CC)C(=O)NC1(C2CCCCN2C(c2cnc(O)s2)=O)CC1 Cc1ccc(O)c(CC(=O)NCC(C)N(C)C(c2cnc(Cl)[nH]2)=O)c1 Cc1cccc(Br)c1C(C(=O)NCBr)NC(=O)C(F)C(C)(C)O.C(C(C)(C)C)=CC=C CC1CC(C)(C(=O)NCCCOCCNC(C2CC2[N+](=O)[O-])=O)CCO1 c1(CN2CCC(NC(c3ccc(CO)o3)=O)CC2)cc2n(n1)CCSC2 CC(C)CC(O)C(C)C(=O)N1CCC(F)(C(=O)NC(c2nccs2)C)CC1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(CNC(=O)Cc2ccccc2)C12CCC2 CCC1=C(C(=O)NOC(CC)C(=O)Nc2ncc(C)cc2OC)CCCO1 C(=O)(CC(O)CC(C)C)N1CCC(C(C(=O)NC(C(=O)NCCC)C)F)C1 N1(C(c2c(C)nns2)=O)CC2(CC(NC(C3SCCCS3)=O)CO2)C1 CCC(C)C(O)CC(=O)NC1CC2(C1)CN(C(C13CCCC(CO1)C3)=O)C2 Cn1nnc(C=CC(N2CCN(CCCCCNC(=O)CCC3CC3)CC2)=O)n1 C(=O)(C(CCC1CC1)NC(=O)Cc1cc(C)on1)NC(c1ccco1)C#C CS(=O)(=O)C=CC(=O)NC1CN(C(c2ccnn2CC(F)F)=O)CC12CC2 c1(SC(C2CCCN(C(=O)NC3CCC3)C2)C)nnc(O)n1C CC(F)(F)CCC(=O)NCC(=O)NCC(N1CCSCC1)=O C1(CCNC(=O)CCc2cc(C)[nH]n2)(NC(C(C2CCCO2)OC)=O)CCCC1 c1(CC(=O)N(C(C2CCCC2)CNC(COC(CC)C)=O)CC)cc(F)ccc1O N1(C(C2(NC(Cn3ccc(C)n3)=O)CCCCC2)=O)CCOCCC1C c1(C(=O)NCC(CNC(c2cc(CO)ccn2)=O)F)cccc2ncccc12 C1(C(C)(C)O)(CNC(C2CC3(CC3)C2)=O)CN(C(=O)C(F)C2CCC2)C1 C1(C(=O)NCCN(C(=O)C(c2ccccc2)C)CCOC)CCC(OC)C1 CCCC(CCC)CC(=O)NC1COC2(CCN(C(c3cccnc3N)=O)C2)C1 C(=O)(CS(=O)(=O)CCO)NC1CN(C(CCN2C(=O)CCC2)=O)CC(O)C1 C1(N(C(CC(C)c2ccco2)=O)C)CN(C(C2CC2C)=O)CC1(C)C n1(CC(=O)N(C2CC(NC(C3ON=C(CC)C3)=O)C2)C)cc([N+](=O)[O-])ccc1=O c1(C(=O)NCC(CO)NC(c2c(C)ncnc2O)=O)cc2c(Cl)cccc2[nH]1 C(=O)(C1=CCCOC1)N1CCCC(NC(C=CC(=O)OC(C)(C)C)=O)C1 C(CC(=O)NCC1(F)CCC(C)(C)C1)(C(F)(F)F)NC(c1ccc(CSC)o1)=O C1(CNC(C(C(C)C)NC(C)=O)=O)CC(C(=O)N2OC3COC23)=NO1 C(=O)(CCC(=O)NC1CC(NC(=O)C(c2cccc(Cl)c2)N(C)C)C1)NC C1=COC(c2ccccn2)N(CC2=NOC3OCCCC23)C1 c1(CC(=O)NC(C)CCNC(=O)CN(C)C2CC2)cc(Cl)c(Br)cc1F N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C(C2CCC(=O)O2)=O)CC(C)(F)C1 Cc1nc(CNC(=O)C(CNC(c2c[nH]c(C(N)=O)c2)=O)CC2CC2)sc1C Cc1ccc(CNC(C2CC(C)CN2C(C2CC2[N+](=O)[O-])=O)=O)nc1 c1(C(N2CC(CNC(CC(CC)SC)=O)C(O)C2)=O)cc(C)c(Cl)cc1F Cn1cnc(C(=O)NC2CCC(CNC(C3(c4ccno4)CC3)=O)C2)n1 N1(C(c2cnc(C)cn2)C(=O)NCCOC)CCCC2(C)CCCC12 c1(C(=O)NCC2N(C(CC(=C)C)=O)CC2)nn(CCOC)c(=O)c2ccccc12 N1(C(CC2C(N(C(=O)CCc3nc(=N)[nH][nH]3)CCC)C2)=O)Cc2ccc(C)cc2C1 c1(CN2CCC(N(CCC)C(c3cc(-c4cccs4)on3)=O)C2)ccc(O)cc1 N1(C(c2c[nH]nc2Cl)=O)CC(O)(n2cc(CC3(Cn4cncn4)CC3)nn2)C1 C1(NC(CC(=O)OC)=O)C2CCC1N(C(=O)Cn1cnnc1O)C2 c1(N)ccc(S(=O)(=O)N2CCN(CCO)CC2)cc1Cl.N=c1[nH][nH]c(=N)c(I)n1 Cc1cc(S(=O)(=O)N2CC3(CC3)CC2C(=O)Nc2c[nH]nc2Br)c(C)cc1Cl C1(OC(C)=O)CN(C(=NCCOCCOC)NCC(C)C)CC12CCC2 N1(C(COC)=O)CCN(C(c2ccc(F)cc2OC)=O)C2CCCCC12 c1(CSCC(=O)NCC(CC)NC(=O)CC2CC2(Cl)Cl)ccc(C#N)cc1 c1(C(N2C(C)CC(CNC(C3CC4CCC(C3)S4)=O)C2)=O)cccc(O)c1Cl c1(NC(C2(F)CCN(C(CCCCC#N)=O)C2)=O)cc(F)c(CO)c(F)c1 CN1CCN(C(=O)C(c2ccc(F)cc2)(F)F)CC1CNC(C1CCCC1)=O Cc1cnc(C(N2CCC(N(C)C(C3COCCC3(F)F)=O)C2)=O)cc1Cl N1(C(C2C(CCC)CN(C(c3ncccc3CC)=O)C2)=O)C(C)CC2CCCC12 N12CCn3ncc(c3C1)C2.CC1CN(CC2CCOC2)CCS1=O.c12cn(nn1)C2 N1(C(CCNC(=O)NCC(CCO)OC)=O)CSCCSC1 Cc1ncc(C=CC(=O)NC(C)CC(C)NC(C23CC(CO2)C3)=O)s1 c1(C(C)C)ncc(C(=O)NC23CC(NC(C4C5CCC45)=O)(C2)C3)[nH]1 N1(C(Cc2scc(CC)n2)=O)CCCC2CN(C(c3ccnc(Cl)c3)=O)CC12 C(=O)(CS(=O)C(F)(F)F)N1CC(C)(NC(C2CC3(C2)CC3(F)F)=O)C1 c1(C(=O)NCC=CCNC(C2(C)CCC(=O)C2)=O)c(F)ccc2n[nH]cc12 C(CCN=c1[nH]c(=NCCc2ccn(C)n2)c2[nH]ccc2[nH]1)N(C(C)C)C CC1(C)CCN(C(C2C3CCC(F)C23)=O)CC1NC(=O)COCC1CCCC1 Cc1c(NC(c2ccncc2-c2nn[nH]n2)=O)cnn1CC(=O)NCC(F)(F)F c1(CC(=O)NCc2cc(C(=O)NCCC(C)CO)no2)c(F)cccc1Cl C1(C(N2CC(OC)(CNC(=O)Cn3cc(C(F)(F)F)nn3)C2)=O)CC1C1CCC1 C1(NC(C2(C(N)=O)CC2)=O)CCC12CCCN(C(=O)CC1(C3CC3)CC1)C2 C1(NC(c2ccc(SC)s2)=O)CCC2(CCN(C(=O)C3=C(C)CCC3)C2)C1 c1(CC(=O)NC(C)(CNC(=O)CCOCC(F)F)C2CC2)cccc2sccc12 c1(C(N2CCC(NC(C(CC)(C)COC)=O)C2)=O)c[nH]c2cccc(Cl)c12 C(=O)(C1=CCCCCC1)NC1(C)CCCN(C(C2CC(=O)C2)=O)C1 c1(OC)cc(Br)cc(C(=O)NCC(C)S(C)=O)c1N Cc1ccc(C(N2CC3CN(C(=O)C=CS(C)=O)CC3(C)C2)=O)c2c1CCC2 N1(C(Cc2ncc(C)o2)=O)CCC2(CCC(NC(c3csc(O)n3)=O)C2)CC1 c1(OC)cc(CN(C)CC2CCCN(C(c3cc(Cl)ncc3C)=O)C2)c(F)cc1F c1(-n2c(CCOC(=O)Cn3cc(CC4CCCO4)nn3)noc2=O)ccc(Cl)cc1 CCC(CCCC(F)(F)F)Nc1cnn(CC(F)(F)F)c(=O)c1Cl N1(Cc2ccc(OCCC#C)cc2)CC(=O)N(CC2CCCC(C(C)C)O2)C1=O c1(CC)ncnc(N2CC3C(NC(=O)COC4CCOCC4)C3C2)c1F C1(C(N(CCNC(c2ccc(NC)c(O)c2)=O)CC)=O)CCCCN1S(N)(=O)=O CCCC(O)C(=O)NCC(N1CCN(C(c2cc(C)n(CC)n2)=O)CC1)C c1(C(N2CC(NC(C(CC)N(C)C)=O)C(C)(C)C2)=O)c(Cl)cccc1[N+](=O)[O-] Cc1noc(N)c1C(=O)NC1CC(OCC(=O)NCc2cnccn2)C1 CC(C)C(O)C(C)(C)C(=O)NCC1CCC(C(=O)NCCCCF)O1 c1(C(=O)NCC(C)CNc2ncncc2Br)c[nH]c2cccc(F)c12 C1(OC)CN2CCCC2(C(=O)N(CC(C)NC(=O)C(C2CCOC2)OC)C)C1 c1(Nc2c(F)c(F)c(F)c(F)c2)cc2ncnn2cn1 n1(CC=CC)ccnc1C=CC(N1CC(C)(NC(=O)CC2COC(C)(C)C2)C1)=O N1(C(=O)Cc2c(F)cccc2Cl)CCC2CCCN(C(=O)C3=COCCO3)C2C1 N1(C(C(C)CO)=O)CC(C2CCN(C(C3CCC4(CC3)CC4)=O)CC2)C1 c1(C(N(CCNC(C2(C#C)CCC2)=O)CCOC)=O)cc(C)n(CCO)n1 C1(CNC(c2ncnc(C)c2Br)=O)(CO)COCC2CCCCN12 Cc1cc(C(N(CC(O)CN(C)C(c2cccc(C3CC3)c2)=O)C)=O)n(C)n1 C1(CNC(C2C(OC)CC2)=O)CCN(C(c2ccc(C)nc2O)=O)CC1(F)F C1(C(=O)NCC2C(NC(COCc3c(C)cccc3)=O)CC2)CC2(CCC2)CO1 C(=O)(C(C)(C)CCC(=O)NCC(O)CN(C)C(C1CC=CC1)=O)OC c1(CC(=O)NCC(CNC(c2cc(C(F)F)[nH]n2)=O)OC)cncn1C C1(NC(c2occ(C)c2C)=O)CC2CN(C(c3ccnc(C(N)=O)c3)=O)CC2C1 C(=O)(CC1=CCOCC1)N1CC(NC(c2n(C)c(S)nc2)=O)C(C(F)F)C1 N1(C(C=CC(c2c(OC)cccc2F)=O)=O)CC(C(F)(F)F)C(S(=O)(=O)N(C)C)C1 c1(C(N2CCSCC2)=O)ccccc1-n1cc(CCC2CCOC2=O)nn1 C1(C(C)C)CN(C(c2sccc2C(N)=O)=O)CCC1NC(=O)CCC(=O)N(C)C C1(NC(c2cc(C)[nH]n2)=O)(CO)CCN(C(c2nc(CC(C)C)sc2C)=O)CC1 N1(C(c2cn(C)nc2)=O)C(C(=O)N(CC(F)F)CCO)CCC12CC2 c1(OCC)ncc(C(=O)NC(CNC(=O)CC2CCCC(C)C2)CCOC)cn1 C1(C(=O)NC2(CC)CC2)CCCC(C(N2CC(OC(C)C)C2)=O)C1 C1(C(C)(C)O)CCN(C(=O)CN2CCC(CN3CCCCC3)C2)C1 c1(C(N2CC(C(C)NC(c3cccc(=O)o3)=O)C2)=O)cc(Cl)cc2cccnc12 Cc1c(C(=O)NC2CC2NC(c2cnn(-c3ccccn3)c2)=O)cccc1F c1(SC)ccc(NC(=O)CN2CCC(N3CCC(CN(C)C)C3)C2=O)cc1 Cc1ncc(NC(=O)CC2(CNC(C3CCCC(=O)CC3)=O)CC2)c(C)n1 c1(CC)noc(C)c1C(=O)NC1CCN(C(C2CCOC(C(C)C)C2)=O)CC1 N1(C(C2(CC#C)CC2)=O)CCN2CCN(C(=O)COC(C)C)CC2C1 N1(C(c2cc(CCC)ncc2)=O)CCC(CNC(c2nccn2CC)=O)C(C)C1 C1(C(N(C)CC2N(C(c3cc(C)sc3)=O)CCC2)=O)CC2(C1)CC21CC1 C1(CNC(c2ccc(SCC)nc2)=O)CN(C(=O)C=Cc2ccco2)CCCO1 N1(C(c2cc(CCC)nn2C)=O)CC2CC1CCC2NC(=O)CNC=O C(CCC(=O)NC1CC(CC(=O)N(C(C)CC(C)C)C)C1)=C(C)C c1(C(N2CC(CNC(C(C(C)C)NS(C)(=O)=O)=O)C(C)C2)=O)cncc2[nH]ccc12 c1(C(=O)NC2CCN(C(C3CNC(=O)N3)=O)C2)cnc(S)n1-c1ccc(F)cc1 C(=O)(C1=C(C)CCCC1(C)C)N1CC(CC)C(NC(c2ccnnc2Cl)=O)CC1 C1(NC(c2scc(CC)n2)=O)CN(Cc2cccnc2Br)CCC1O N1(CC(=O)NC(CCC)=O)CC(C)(CNC(=O)CCc2nccs2)C1 Cc1ccc2c(c1)SC(C(N1CC3CN(C(=O)C(C)n4ccnc4)CC3C1)=O)C2 N1(C(CCC=C(C)C)=O)CCCN(C(c2cc(C(F)F)cs2)=O)C(C)C1 C1(OC(CN(C(C)(C)C)C(C2C(C(=O)NC)C2)=O)=O)CCSCC1 C1(C(=O)NC2CCCC(CC)C2)CCN(C(=O)c2nnc(S)n2C)O1 N1(C(C(C(C)C)n2cccc2)=O)CCCOC(CNC(=O)C(O)C2CC2)C1 C(=O)(CCS(=O)(=O)C1CCCC1)NC12C(CN(C(CCC(=O)NC)=O)C1)CCC2 c1(NC(CN(C(CCN(CC)CC)=O)C)C)ncnc2sc3ccccc3c12 C1(C(C)C)CN(C(c2cnc[nH]2)=O)CCN1C(C1CC(OC(F)F)C1)=O c1(C(N(CC(N2CCC(O)(CC#C)CC2)=O)CC(C)C)=O)ccc2cc[nH]c2n1 C1(CCNC(CC(=O)NCC)=O)CN(C(=O)CCn2cc(Br)cn2)CC(C)O1 C1(C(N2CC(CNC(C3=NNC(=O)CC3)=O)OCC2)=O)CCc2nncn2CC1 c1(NC(C)Cc2ccccc2O)ccc(N2CCSCC2)c(Cl)c1 C1(NC(c2c(C(C)C)ncs2)=O)CCN(C(=O)C(F)C2CC2)CC(C)(C)C1 C(C(=O)NCCC1(CNC(c2nn(C)cc2C(C)=O)=O)CC1)(C(C)(C)C)OC c1(CN(C(C(C(C)C)SC)=O)C)ccc(Cl)cc1Cl c1(C(=O)NC(C(CCC)C)COC)c(O)cccc1[N+](=O)[O-] N1(C(C(C2CCN(C(c3ncnc(C)c3C)=O)C2)C)=O)CCc2n[nH]cc2C1 c1(CC(=O)NC2(CNC(=O)CC34CCCC3C4)CCCC2)c(O)ncnc1O c1(C(C(=O)NCC(CNC(C2(CC=C)CC=CC2)=O)O)OC)cccc(OCC)c1 C12(C(=O)NCc3c(C4CN(C(C(C=CCCC)O)=O)C4)ocn3)CCC(OC)C1C2 CCCCCC(O)CC(=O)N1CCN(C(C)C(=O)NCc2ccccc2C)CC1 CCCCC(C)(F)C(=O)N1CC=C(C(=O)NCC(C)(C)CCO)C1 CC(=O)CCCC(=O)N1CCC(O)(C(C)NC(c2nccc(Cl)c2F)=O)C1 CCC(C)(CNC(=O)CCC1CCCCC1)C(=O)NC1CC(CO)C12CCC2 C#Cc1cc(C(=O)NC(C)C(C)C(=O)N2CCC2(C)C)ccc1C C12(C(N3CCC(O)C3c3ccccc3Cl)=O)CC(CC1CO)C2 N1(C(CCC=C(C)C)=O)CC2CC(C1)N(C(=O)C=Cc1cscn1)C2 C(=O)(C#CC1CCOC1)NC(C(C(=O)Nc1c(OC)ccc(O)c1)C)C Cc1nc(CNC(=O)C(O)CN(C)C)oc1C(=O)NC1(C)CCOC1 N1(CC(C)(C)NC(C(CC)O)=O)CCN(C(=O)CC2CCCN2C)CC1 CC(C)CS(=O)(=O)CC(=O)N1CC2CCCC(NC(=O)Cc3ccccc3)C2C1 N1(CCCC)CC=C(CNC(=O)CN2C(C)CCC2C)CC1 c1(OC)cc(C(N2CCC3CN(C(c4ccccc4F)=O)CC23)=O)cc(O)c1O C1(NC(c2ccoc2)C)CCN(C(=O)CC2CC(C)(C)C2)CC1C C1(C(=O)NCC2(C)CCN(C(=O)CCC3(O)CCC3)C2)COc2ccccc2O1 CCC(C)C(C(=O)NCCCC(C)C)N(C)C(c1ccccc1)=O CCCC(C)(O)C(=O)N1CC(O)(c2cn(CCC3CC(C(C)C)=NO3)nn2)C1 CCCCCCCCCC=CC(N1CC(NC(=O)C(C)C2CCCC2)C(F)C1)=O C1(CNC(C(C)O)=O)CN(C(c2ccc3c(c2)CCC3)=O)C2COCC2O1 C1(C(=O)NC2CN(C)C(C)(C)C2)(CC)CCN(C(C2CC(=C3CCC3)C2)=O)CC1 C(CC(C)(C)C(=O)NCC(C)CN(C)C(c1cc(C)ncc1C)=O)OC N1(C(c2c(C)nsc2)=O)CCC2(CC1)CC2C(=O)NCc1sccc1Cl N1(C(CCC(=C)Cl)=O)CCCC(CCNC(=O)C(C)(C)CCF)CC1 N1(C(c2ncccn2)=O)CCCC2(CCCN2C(=O)CC2CCCC2)C1 c1(OCCC(=O)N(C2CN(C(C3C(SC)CCC3)=O)C2)C)ccc(C)cc1C C1(c2cn(CCC=C)nn2)CCN(C(c2cscc2C)=O)CC1 C12CCN(C1)C(=O)N2C.n1(C(C)C(=O)OC)cc(CC(c2ccccc2)=O)nn1 N1(C(c2ccc(CC)cc2)=O)CCC(NC(=O)COC)C(CO)C1 C1(CNC(C(CC=C)(C)CC)=O)CCCC2CN(C(=O)Cc3cc(C)[nH]n3)CC12 C1(CNC(=O)NCCc2cnc[nH]2)CC2(C1)CC21CCC1 C(=O)(CC1=CCCCC1)N(C)CC1CCN(C(c2c(CC)c[nH]n2)=O)C1 C12(NC(CCCOCC)=O)CCCC1CN(C(=O)CCc1nc(CSC)no1)C2 c1(C(=O)OC(c2onc(CCC)n2)C)cc(Br)ccc1Br c1(C2C(C(N3CC(CS(N)(=O)=O)C3)=O)C2)ccc(Br)cc1F C1(C(=O)OC)COCCN1C(C1CC(NC(=O)CCc2ccsc2)C1)=O Cc1cc(C(=O)NC2(CC(O)CO)CC2)c(C)n1C1CCCC1 Cc1ccc(CC(=O)NCC2(O)CCCN(C(=O)CC(C)(C)O)C2)cc1Cl Cc1ccc(F)cc1C(N1CCOC(CC(=O)NCC(C)(F)F)C1)=O c1(CC(=O)OCC)c[nH]c2ccc(OC(C3COC(C)(CCCOC)O3)=O)cc12 C1(C(N2CC(F)(CNC(C3(C)ON=C(C)C3)=O)C2)=O)CCc2cncn2C1 N1(C(c2cc(CNC(C3(C=C)CCC3)=O)nn2C)=O)CC2(C1)CC(C)(O)C2 C(=O)(CC(C)CCC(=O)NC1CC(C)CN(C(=O)C2=C(C)OCCS2)C1)OC C12(C(=O)NCC(C)(C)NC(C(CC#C)CC#C)=O)CCC(CC1)C(C)(C)O2 c1(CC(=O)NCC(CC)NC(C2(SCCl)CC2)=O)ccc(OC(C)C)cc1.C(C)(C)O C1(C)(NC(C(CC(C)C)NC(=O)CC2CC3C=CC2C3)=O)CC(C)(C)OC1=O c12c(OC)ccnc1c2=O.C12(NC(c3cn(CC)nn3)=O)COC(CNC)(C1)C2 C1(CNC(c2nn(C)c(C(N)=O)c2)=O)CCC(C)(C)CN1C(c1ccoc1)=O N1(C(CC=C(C)C)=O)CC2CN(C(=O)Cc3cccnc3C)CC(F)(F)C2C1 c1(NC)cnc(Cl)cc1C(=O)NCC1CN(C(c2cnc(Cl)[nH]2)=O)CCO1 c1(SC)nncn1-c1ccccn1.C(C(=O)NCCO)N(CCOCC)C C1(N(CCO)CC)CCCN(C(c2ccnn2C(C(=O)NC)OC)=O)C1 C1(NC(=O)CCc2cccnc2)C2CN(C(=O)C(c3ccc(F)cc3)F)CC12 Cc1[nH]nc2c1CC(C(N1CCC(CCNC(C3(C(N)=O)CCC3)=O)C1)=O)CC2 C1(C)(CNC(C=C(CCC)C)=O)CCN(C(c2cc(N(C)C)nc(Cl)c2)=O)CC1 N1(C(C2C(c3ccc(C)o3)C2)=O)CC(C2CN(C(c3ccc(Br)cc3)=O)C2)C1 C1(C(N(C2CCN(C(C3CN(C(C)=O)C3)=O)CC2)CC)=O)OC2CCC1CC2 n1(CC#CCC)c(-c2cnn(C)c2)csc1=Nc1cnn(C)c1 c1(CC(=O)NCC(C)N(C(=O)CCc2cn(C)cn2)C)cncnc1O C(=O)(CCCCCO)Nc1cccc(NC(CC(C)(F)F)=O)c1 Cc1csc(C(=O)NC2CC(O)C2CC(=O)N)c1.c1(C2(C)CC2)ncccn1 C1(CNc2cc(C)c(-n3ccnc3)cc2)CC(C)N(C)CC1C CC(CCNC(=O)CCCNC(N)=O)CCNC(c1cnc(CC(C)(C)C)s1)=O C1(C(=O)NCC2C(C)(C)C2(C)C)CC12CCN(C(C1CCCCC(=O)C1)=O)CC2 CC(C)C(C)(O)CNC(=O)CCC1CCC(NC(=O)C(C)(C)CO)C1 N1(C(=O)CO)CCN(C(=O)CNc2cnc(CC)[nH]2)CC1CC(=O)OC N1(C(CC(COC)NC(=O)CCC2CC2(C)C)=O)CCCC2(CCOC2)C1 N1(C(c2c(OC)scc2)=O)CCCC2(CCN(C(=O)C(O)CC(C)C)CC2)C1 C1(NC(c2ccc(CNC(COCCOC)=O)o2)=O)CC2CCC2C1 c1(C2C(C(N(C3CCC(O)CC3)C)=O)C2)cc(F)cc(Cl)c1 CC(O)C(C)(C)C(=O)NCC1(NC(c2cc(CCO)on2)=O)CCCC1 C(C(F)(F)F)(NC(=O)NCCCc1onc(C(C)OCC)n1)SC CN1CCCC(F)(C(=O)NCC2CN(C(c3c[nH]c(=S)cn3)=O)C2)C1 c1(NC(C)C)ncc(C(=O)NC(C)(CNC(=O)CC2CCC2)C2CCC2)cc1Cl c1(CN2CCC(O)(C(=O)NC(c3c(C)nc(OC)s3)C)C2)c(O)cc(O)cc1O c1(C(C(=O)NCCCC2CC2)N(C2CCC2)CC)ccsc1C N1(C(C2CCc3ccnn3C2)=O)CCC2(CC1)CCN(C(C1CCO1)=O)CC2 c1(NC(Cn2c(=N)nc[nH]2)=O)nc2cc(OCC(F)(F)F)ccc2s1 c1(OC)cc(CN(CCO)CSC(C)C(=O)O)ccc1OCc1cccnc1 C1(C(=O)NC(C=C)COC)C2CCCC2CN1C(=O)C(C#N)C(C)(C)C CC(C)(C)CCCC(=O)NCC1(C(=O)NC2CCC3CC2CO3)CC1 C=C1CCN(C(=O)CCC=CC)C(C(=O)N(CC(O)COC)C(C)C)C1 Cc1ccc(NC(=O)CC2(N(C(=O)C#CC3CC3)C)CC2)cc1C C(=O)(C(C)(O)C(C)C)N1CC(NC(C(n2c(C)ccn2)C)=O)C(O)C1 C(=O)(CN=S(C)(C)=O)N1CCC(CNC(C(C)NC(c2ccc(N)cc2)=O)=O)C1 C1(N(C(c2cc(Cl)c[nH]2)=O)CC)CCCN(C(=O)Cc2ccccc2F)CC1 c1(SCCNC(N2CCC(N3CC(O)C3)C2)=O)ccc2c(c1)OCO2 O=C1CCc2ccc(C(=O)NC3CC(NC(C4CC4F)=O)C3)cc2CN1 N1(C(C2N=C(C)SC2)=O)CCN(C)C(CNC(c2ccc(NC(N)=O)cc2)=O)C1 C=CCCCCCCC(=O)N1CCCC(C)(C)C1C(=O)N(C1CCC1O)CC C1(C(N(CC)CC2CC(=C)C2)=O)CCN(C(=O)Cn2ccnc2C)C1C c1(SCC=CC(=O)NCC(C)N(C)C(c2cnn(CC(F)F)n2)=O)ccccn1 C(CCC(C(=O)NC1CC(O)C1OC)NC(c1ccc(C)cc1O)=O)OC C(C1c2ccccc2CN1C(c1cc(Cl)ncc1N)=O)NC(CCC(C)OC)=O C12(NC(c3nc(N(C)C)oc3)=O)CCOC(CNC(C3(O)CCCCC3)=O)(C1)C2 CC(C)(C(=O)NCC(C)(O)CNC(c1c[nH]nc1-c1ccncc1)=O)C1CC1 C1(CC(=O)NCc2cc(C)oc2)CCCCC1NC(c1nccnc1N)=O c1(C(N2CC(O)(CN(C)C(C3CCOC3)=O)C2)=O)cc(Br)n2c1CCC2 C1(C)(CC(=O)NCC(c2cccs2)C)CCN(C(c2ccccc2C2CC2)=O)C1 C1(c2n(CCSC)nnn2)(NCc2csc(C(F)F)n2)CCCC1N1CCCC1 Cc1cc(CC(N2CCCC2C(C)(C)NC(=O)CC23CC(C2)C3)=O)n[nH]1 C1(CCCOC)CN(C(C2CCC(CO)CC2)=O)CCO1.C12CCN(C1)C2 c1(C(=O)NCC(CNC(C(C)C(C)(C)C)=O)O)csc2c(Cl)cccc12 c1(C(N2C3CN(C(Cc4n[nH]c(=NC)s4)=O)C(CC3)C2)=O)ccc([N+](=O)[O-])cc1F CCC(O)C(C)(C)C(=O)NCc1ccoc1C(=O)N(C1CC(F)(F)C1)C Cc1nc(C)c(C(=O)NC2COCCN(C(C3(N=[N+]=[N-])CC3)=O)C2)nc1C C(=O)(C(C)CC(N)=O)NC1(c2ccccc2)CN(C(C=Cc2ccc(C)s2)=O)C1 CN1CCCC2(CCN(Cc3conc3C3CC3)C2)C1=O C1(N)C2CN(C(=O)Cc3cccc(OC)c3)CC12.C12(C(=O)OC)CC(C(=O)OC)(C1)C2 CC(CN=c1[nH]n(C)cc1[N+](=O)[O-])NC(=O)CC1CCCCO1 C(=O)(C(O)C(C(C)C)OC)NC1(c2cc[nH]n2)CC1.C(CCC(=O)NC)OC C1(NC(=O)NC2(c3n(C)ncc3)CC2)CS(=O)(=O)C12CCCCC2 Cc1ccc(C(N2CCC(O)C2C(=O)Nc2ncccc2CO)=O)c(C)c1F c1(C(=O)NCC2CN(C(C3C(C)(C(=O)OCC)C3)=O)C2)cc([N+](=O)[O-])c(C)s1 C(=O)(C(F)CCC(C)(C)C)NCC(C)N(C(CCCOCCOC)=O)CC CC1(C)CCc2sc(NC(=O)NC34CC3CS(=O)(=O)C4)nc21 CN1CCOC(C(=O)N(C)CC2CCCN(C(=O)CC(=O)OC(C)(C)C)C2)C1=O C(C(CC(=O)NC(CC1CC1)CO)NC(c1cnc(N)cn1)=O)OC CC1CC(NC(c2cnnn2C2CC2)=O)CN(C(=O)C(C2CCCCC2)O)C1 c1(C(=O)NCC(CNC(c2ccsc2F)=O)CO)ccn2cnnc2c1 C=CC1OCCC1C(=O)NC(C(=O)NCCNC(=O)NC(C)C)C1CCCC1 c1(CC)ccc(OCC(=O)N(C)CCNC(=O)CC2CC2)cc1 Cc1ccc(F)cc1C1CC1C(=O)NCC1(NC(c2cscn2)=O)CCCCC1C c1(C(=O)NCC2CCN(C(CC(C=C)CC)=O)CC2O)c(Cl)ccc2c1OCO2 c1(C(=O)NC2CC3(CN(C(C(CC(C)C)F)=O)C3)C2)cc(F)c(F)cc1Br C12(C(=O)NC3CCCC(NC(=O)COc4cn[nH]c4)C3)CC3CC(C(=O)N1)C2C3 CCC(C(=O)N1CCCCC(C(=O)NC(C)(C)CCN(C)C)C1)C(C)C C1(NC(C2CC(C)C2)=O)CN(C(=O)C=CC2CCC2)CC1c1cccc(F)c1 C1(NC(COCC=C)=O)CN(C(c2cscc2C(F)(F)F)=O)CC(C)(C)C1 C(C(=O)NCC12CC(NC(=O)C(C)CN(C)C)(CO1)C2)(C(C)C)SCC n1(C(=O)Nc2nnc(N3CCC(OC)CC3)n2C)ncc(C#N)c1I C(=O)(C(C(=O)NCCN1CCC(NC(=O)CCC2CC2)CC1)C(C)(C)C)OCC Cc1nn(C)c(Cl)c1C=CC(N1CC(NC(=O)C=Cc2cnccn2)C1)=O Cc1ccccc1OCCCC(=O)NC1COCC1NC(=O)CN(C)C(C)C c1(CC)cc(C(=O)N(C)CC2CCCCN2C(c2ccc(Cl)s2)=O)ncn1 C1(c2n(C)ccn2)CN(C(=O)C(C)(C)c2ccns2)CCN1C(C1CCCO1)=O N1(C(C2(C(N)=O)CC2)=O)CC2(CCCC(CNC(=O)CC3CC=CC3)O2)C1 N1(C(c2[nH]cc(CC)c2)=O)CCC2(C1)CN(C(=O)CC(C)(C)SC)CC(C)O2 C12(NC(CCC3OCC(C)(C)C3)=O)CCC(NC(=O)CC3CC3(Cl)Cl)(CC1)C2 c1(OC)cc(C)c(NC(C2CC2C2CN(C(c3csc(=N)[nH]3)=O)C2)=O)cn1 C1(C(=O)NCC(N)=O)CCCN1NC(=O)C=CCF.CON(C)C(=O)C c1(C(=O)NCCC2CCN(C(c3cc(CC)c(C)s3)=O)C2)cc(C)n(CC)c1C C1(CNC(c2nn(C)c(=O)cc2)=O)CN(C(c2cncc(Cl)c2)=O)CC(C)(C)C1 Cc1ccc(F)cc1CC(C(N1CCN(c2nc(C3CCCC3)ns2)CC1)=O)C C1(CNC(c2n[nH]cc2Cl)=O)CCCN(C(C2CCCN2CC(F)(F)F)=O)CC1 C(=O)(C1=NNC(=O)CC1)N1C(CCNC(C(CC=C)NC(C)=O)=O)C(C)CCC1 N1(C(CCOCCOCC)=O)CCC(CNC(=O)COC)(OC)C1 Cc1cc(C(C)NC(=O)C(=O)NCCCc2cn(C3CC3)nn2)cc(C)c1I C1(NC(=O)C=Cc2cccs2)CCN(C(c2cnc(C3CC3)nc2)=O)CC(O)C1 N1(C(C2(C#C)CC2)=O)CCC(C(C)CNC(c2onnc2CC)=O)CC1 c1(C(N2C(CC)C(NC(c3ccsc3)=O)CC2)=O)cc(=O)n2nccc2[nH]1 C1(C)(C(=O)NC2CCN(CC)C(C)C2)CN(C(C2CC2CC)=O)C(C)(C)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CCC(O)(CN(C)C(c2ccsc2C)=O)C1 N1(C(C(=O)N(C)C)=O)CCC2(CC2NC(c2cnc(C(N)=O)cn2)=O)C1 c1(CC(=O)N(CCCNC(C2CC2CF)=O)CCO)c[nH]c2ccccc12 C1(C2CC2)(NC(C2ON=C(CC)C2)=O)CCN(C(=O)Cc2cc(C)on2)C1 C#Cc1ccc(C(=O)NCCCOCCCNC(C2C=CCS2)=O)cc1 c1(C(=O)NC2CN(C(=O)CC3CCCCO3)C2)cnc2[nH]cncc1-2 c1(CC(N2CCC(F)(F)C(CNCC34CC(C3)C4)C2)=O)cccc2occc12 C12(C(N3CC(OC)C3)=O)CC(CCO1)N(C(C1CC(=O)CCO1)=O)C2 N1(C(CN(C)C)=O)CCCC(O)(CCNC(C23CC(C)(CO2)C3)=O)C1 c1(CNC(=O)NC2CN(C(=O)C(=O)NCC(F)(F)F)C2)ccnc(F)c1F c12ccccc1ON(C(C)C1CC1)CCC2.c1(CC)nc(-c2ccccc2)no1 C1(Nc2c(C(=O)OCC)cncc2)CCC2(CC1)CN(C(=O)C(C)(O)C(C)C)C2 N1(C(CC2=C(C)CC2)=O)CCN(C(c2ccnn2C(C)C)=O)CC2CCCCC12 C(C(C)CN=c1cc[nH]c(C#N)n1)N1CCN(C(C(=C)C(F)(F)F)=O)CC1 N1(C(c2cnc(OC)s2)=O)CCCC(C2CN(C(=O)C=C3CCC3)C2)C1 N1(C(c2cc(CC)on2)=O)CCC=CC1C(=O)NC(C)C(CC)CC Cn1cc(S(N)(=O)=O)cc1CC(=O)NC1CC1NC(c1c(Cl)ccc(O)c1N)=O c1(C(N2CCN(Cc3c(C)n[nH]c3C)C(CC#N)C2)=O)cccc2ccoc12 C1(C(=O)NCC2N(C(CCC(C)c3ccccc3)=O)CC2)CCOCC12CCC2 C=C=CC(C)C(=O)NCCC1COCCN1C(c1cc(C(=O)OC)co1)=O c1(CC(C(=O)NC(C)C2CC2)NC(=O)NC(N)=O)cnn(C)c1O c1(C(=O)NCCC2CN(C(CC3(C)CCC3)=O)C2)cc(C(F)(F)F)c(Cl)cn1 C1(NC(c2ccc(CO)cc2)=O)CC12CCC(NC(c1ncccc1C)=O)CC2 CN1CC2(CCN(C(C3CN(C(c4ccc5cc[nH]c5c4)=O)CCN3)=O)CC2)C1 CC1CN2CCN1CC2C(N1CCC(CCNC(=O)CSc2ccncc2)C1)=O C1(C(N2CCC(C(C(=O)NC3CC(CSC)C3)C)C2)=O)C2CCC(C2)C1C C1(CNC(C2(CCC)CCC2)=O)COCC1NC(C1CNC(=O)C1)=O CC(C)CC(O)C(=O)N1CC2(CC2)CC1C(=O)Nc1c(Cl)cnn1C C1(N(C(C2(c3nc(C)[nH]n3)CCC2)=O)C)CCCN(C(=O)CN(C)C2CC2)C1 N1(C(C2N(CC)CCCC2)=O)CC2CC(NC(C3CC(=O)N(C(C)C)C3)=O)C2C1 C1(C(C)C(=O)NC(C(F)(F)F)C2CCCCC2)CCC(F)(F)CC1 c1(CC(=O)N(C2CCN(c3ncncc3F)C2)C)ccc(F)c(Br)c1 c1(C(=O)OCC)cc(NC(c2cc(Cl)c(Br)c(Cl)c2O)=O)c2cc[nH]c2c1 C(C(=O)N=c1cc[nH]cc1-c1ccccc1)N(C)Cc1cccc(Br)c1 C1(CC(=O)NC(C)CN(C)Cc2ccc(CN(C)C)o2)(N(C)C)CCCC1 C=Cn1ncc(C(N2CC(O)(C(F)C(=O)NC(C)CC3(O)CCC3)C2)=O)c1N C(=O)(C(C)(C)CC(C)C)N1CC(C)CC(CNC(CCN(CCC)C)=O)C1 CC1(C)Cc2ccccc2C1NCc1n[nH]cc1Br CC1CN(C(c2csc(C(F)(F)F)n2)=O)C(C)CN1C(=O)COCCCN=[N+]=[N-] c1(C(=O)NC(C(=O)N2CC(C(C)(C)C)C2)C(C)(C)O)nccc2[nH]ccc12 c1(CC=C)ccc(C(=O)OCCCOc2cccc(N(C)C)c2)cc1C(=O)OC C(CCC(C)C(=O)N1CCCC(c2ccccc2)(C(=O)O)C1)OC C(=O)(CC1OCc2ccccc21)NCCC(C)NC(C(COC)O)=O C(c1nccs1)=CC(=O)NC1CC(CNC(C2(CF)CCC2)=O)C1 CCCC(C)CN=c1cc[nH]cc1S(=O)(=O)N1CC2C(C(=O)OC)C2C1 N1(CCCCC(=O)NCC(=O)OCC(CCC=C)O)C(=O)c2ccccc2C1=O N1(C(CN(C)CC)=O)CC(CNC(c2cc(CSC)c(C)s2)=O)C2(CCC2)C1 c1(C(=O)NC(C)CCNC(=O)C(C)N(C)C)c(F)ccc2c1OCO2 c1(CNC(=O)NCC2(OCC)CCOC2)ccnc(C2CCCC2)n1 c1(C(N2C(C)CC(CNC(=O)CNS(C)(=O)=O)C2)=O)cccc2cnsc12 c1(OC)c(C(=O)NCCCCN(C)C(C2CC23CC3)=O)occc1=O C1(CNc2c(C)cc(F)c(Br)c2)(CO)COCC2CCCN12 CCCCC(O)CNC(=O)C(c1cnn(C)c1)NC(c1ncoc1C)=O C1(CNC(CC=CCCCCC)=O)CC(C)N(C(c2ccnn2C)=O)C1 S1(=O)(=O)c2cccc(c2)N1.c1(SC)cccc(C(=O)OCC2CC2)c1 C(C(=O)NC1(CC(=O)N(C)CCc2cnccn2)CC1)(C(C)C)OCC C1(O)(CNC(C2(N(C(c3cnn(C)n3)=O)C3CC3)CCC2)=O)CCOCC1 C1(NC(COCC)=O)C2COCC1CN(C(c1n[nH]c(C)c1Br)=O)C2 Cn1ncc(C(=O)NCCNC(c2cc(-c3ccccn3)no2)=O)c1N N1(C(c2ccccc2S)=O)CCC2CN(Cc3ccc(Br)cc3Br)CC12 c1(CC)cccc(C)c1C(=O)NC1(C)CC(NC(c2ccnc(SCC)c2)=O)C1 N1(C(CC(=O)NCC)=O)CCOC(CCCNC(C2(C)CS(=O)(=O)C2)=O)C1 C1(CC)CCCN(C(=O)Nc2cccc(CN3CCCCC3=O)c2)C1 c1(CC(=O)N(CC(C)NC(c2ccc(Cl)c(O)c2N)=O)C)c[nH]c2ncccc12 c1(C(=O)NC(C)CCNC(=O)CC2CC(C)(C)C2)cc(Cl)cc(Br)c1 CC1=C(C(=O)N2CC3(CCCC3NC(=O)C(C)C(C)O)C2)Cn2nnnc2N1C Cc1nc(C(N2CCCC2CNC(C2CC23CCOCC3)=O)=O)c2ccnc-2[nH]1 CC1CCCN(C(C2OCC2(C)C)=O)C1CNC(c1nc(=O)cc(N)[nH]1)=O c1(SCC(=O)NCc2scc(CNC(C(CC)(C)O)=O)n2)nc(C)cc(C)n1 Cc1ccccc1C(C(C)C)N(CCC(=O)O)CC(=O)NC(C)C Cc1nc(C(C)C)ccc1C(=O)NCCCCC(C)(C)NC(c1nsnc1O)=O Cc1c(NC(=O)N(C)C)cccc1C(N1CCC(Sc2ccccc2)C1)=O c1(N2C(C(=O)NCCOCCNC(C)=O)CC(OC)C2)ncnc2cnn(C)c12 N1(C(C(CC)O)=O)CCC(C(C)NC(=O)CCn2c(C)ccc2C)CC1 CC(C)(O)C#CC(=O)N1CCC(CF)(NC(c2coc(CC3CC3)n2)=O)C1 N1(C(c2cc(Cl)ccc2Cl)C(N)=O)CCOC2(CCCC2)C1 C(=O)(CC1=NNC(=O)C1)N1CCC(CN(C(=O)C(CN(C)C)N(C)C)C)C1 c1(C(=O)NCC2CN(C(CC(C=C)C)=O)C2)c(F)cc(O)cc1F c1(C(C2(C)CC2)NC(c2n(CC=C)nnn2)C(C)CC)cccc(Cl)c1 c1(CCC(N2CC(CNC(C=CC=CC)=O)C(O)C2)=O)cccc(OC)c1F n1(CCOCC)cnnc1CNC(=O)C(c1ccc(C)s1)N(C)CCC1CCC1 N1(C(c2c(C#C)cccc2)=O)CCc2ccc(C(=O)OCC)cc2C1.C1(=O)CN1 c1(C(N2CCC3(C(NC(C(CC(N)=O)O)=O)C3)CC2)=O)csc2c(F)cccc12 N1(C(c2cnc(C)nc2)=O)CCCCC(CNC(C2CC(C(C)C)C2)=O)C1 N1(CC(C)Oc2cccc(OC)c2OC)CC(=O)N(CC(C)C)C(=O)C1 N1(C(C(C=C)O)=O)CCC2(CCCN(c3cc4nnc(CC)n4cn3)C2)C1 C1(C(=O)NCCN(C)C(C2(c3ccccc3)CC2)=O)CCC12CCCO2 CC1(C(=O)NCCN2CCC(NC(=O)CCC3CC3(F)F)CC2)CCC[SH]1(=O)[O-] c1(NC(CNC(=O)NC(c2ccccc2)C)=O)cc(I)c(Br)cc1Cl N1(C(COCC(=C)C)=O)CCN(C(c2ccc(C(N)=O)o2)=O)C2CC12 C1(C)(OC)CCCN(C(c2csc(CNC(=O)CC3CCC(=O)N3)c2)=O)C1 C#CC1COCCN1C(=O)C(CCN(C)C)NC(c1cnn(C)c1OC)=O c1(OC)ccc(C(F)(F)F)cc1C(N1CCC1(C)C(=O)Nc1onc(C)c1C)=O Cc1ccc(NC(=O)CC2CCCC(O)C2)c(-n2cc(-c3cscn3)nn2)c1 O=C1CCC(NC(=O)CNC2CCN(C(c3occc3-c3ccccc3)=O)C2)C1 Cc1cnc(N(Cc2ccsc2)CC2CC2)c(S(=O)(=O)N2CCCCC2C(C)C)c1 c1(C(C(=O)NCCCC)N(CC(F)Br)C)ccc2nc(C)[nH]c2c1 C1(c2cn(C)nn2)COCCN1C(c1cc(Cl)cn1CC)=O.CCC(C)C=O CCC(CNC(=O)C(Cc1cc[nH]n1)NC(c1ccnnc1C)=O)(CC)C(N)=O N1(C(CCOC2CN(C(C3(C#N)CC=CC3)=O)C2)=O)CC2CCCC(C2)C1 Cc1c(N)ccc(C(=O)NC2CCCC(NC(=O)Cn3ncnn3)C2)c1C C(CS(=O)(=O)Cc1cn(CCO)nn1)C(=O)NC(c1nc(C(F)(F)F)cs1)CC N1(C(c2cccc(-c3cnco3)c2)C(=O)NCC)CCCC(N=[N+]=[N-])CC1 O=C(CCCO)NNC(=O)C(F)(F)c1c(F)cccc1F N1(C(c2c(CC=C)cccc2)=O)CCC2(CCN(C(C3CC3C)=O)C2)C1 CC1(C)CCC(N=[N+]=[N-])CN1C(CC1CCCCO1)C(=O)NC1CCCCC1 C1(NC(CCNC(=O)NC)=O)CCC(C)(CNC(=O)Cc2ncoc2C)C1 c1(OC)c(F)cc(F)c(CN2CC3(CC3)CC2C(=O)N=c2[nH][nH]cc2I)c1F C1(C2(NC(C3CCN(C(=O)C4(C)CC(=O)N(C)C4)O3)=O)CC2)(OC)CCC1 C=CCCCCCCC(=O)NCC1CC(C)N(C(c2cc3n(n2)CCCC3)=O)C1 C1(C)(CNC(c2cc(C)on2)=O)COCCN(C(C2CC2c2cnn(C)c2)=O)C1 C12(C(N3CCCN(C(C4(CC)CCC(O)CC4)=O)CC3)=O)CCCCC1OCC2 N1(C(Cn2c(C)ccn2)=O)CC2(CCC(CNC(C3CC(C)(C)CCO3)=O)O2)C1 Cn1c(C(=O)NC2CC(CNC(=O)CCc3nc(C(F)(F)F)n[nH]3)C2)nnc1S C1(CNC(c2ncc(OC)cc2F)=O)CCC2(CCN(C(=O)CC3CC3)CC2)O1 Cc1nnc2ccc(C(=O)NC3CN(C(=O)C(C)C)CC3C(F)F)cc2c1C C1(C(=O)NCC(CN(C(=O)CNC(=O)C(F)(F)F)CC)(C)C)CC(=O)OC1(C)C c1(C(=O)NCCOCCn2cc(-c3c(COC)[nH]nn3)nn2)cc2cnn(C)c2s1 c1(SC)snnc1C(=O)NC(c1ccccc1)C1CCC1CN N1(CC(=O)NCCC2CC(NC(=O)CCN3CCOC3=O)C2)CC(=O)NC1=O CCCC(CCNC(=O)C(C1CC1)N(C)C(c1nocc1C(C)C)=O)CCC c1(C(=O)NC2C(NC(c3cnc(CC)[nH]3)=O)CS(=O)(=O)C2)cc2n(c1)CCCC2 N1(C(c2cnc(CC(C)C)s2)=O)CCN(C(c2cnn(C)c2)=O)C(CC(F)F)C1 c1(C(N(CCNC(C(C)c2ccco2)=O)Cc2ccccc2)=O)cc(Cl)no1 c1(CNC(C(CCOC)(C)C)c2nnnn2CCSC)ccc(C)c(F)c1F N1(C(C)C)CCOC(C(=O)NCC2CCC(NC(c3cnc(S)[nH]3)=O)C2)C1 Cc1noc(C)c1CCNC(C1(NC(C2CC(OC)C2)=O)CCSC1)=O CCC(CC(=O)NCC1CCCN1C(=O)CCCc1ccc(F)cc1)C1CCC1 c1(C(N2C(C(C)NC(C3(C)CC3(F)F)=O)CCC2)=O)ccc2c(c1)CCC2(F)F N1(CC(C)C)CCC(C(=O)N(CC(C)CN(C(=O)CC#N)C)C2CCCC2)CC1 C1(CCNC(C(C)=CC)=O)CN(C(=O)C(C)(C)COC(C)C)CC(C)O1 C1(NC(C2CCCN(C(=O)NCCC)C2)=O)CC(C)CN(C(=O)CC(F)(F)F)C1 c1(C(=O)NCC(C)N(C(CC(OC)OCC)=O)CC)ccc(F)c(C(F)(F)F)c1 N1(C(C2(N(C)C)CCC2)=O)CCC(NC(=O)CCC2CCOC2)C(CO)C1 c1(C(=O)NCC2(F)CCN(C(=O)C[SH](CC(F)F)CC)C2)cc(Cl)ccc1C(F)F CC(N=c1nc2c(cnn2C)c(NCCCc2cnn(C)c2)[nH]1)C1CCCCC1 c1(C(N2CC(NC(C(CCC)OC)=O)C(C)C2)=O)cc(=O)c2ccccc2n1C c1(C(N2C(C(N(CCC(C)C)CC(C)C)=O)CC(C)C2)=O)nccc2[nH]ccc12 C1(NC(c2csc(Br)n2)=O)CCSC12CN(C(c1csc(O)n1)=O)C2 CC1CCC(CC(=O)NCC2(F)CC(CNC(c3cn(C4CC4)nn3)=O)C2)O1 C1(CNC(CN(C(COC)=O)C)=O)(NC(C2CC2(F)Cl)=O)CC2CCC1CC2 c1(C(N2CC(N(C(C=C(C)C)=O)C)C2)=O)cc(N2CCCC2)ncn1 N1(C(c2c(C)c[nH]n2)C(=O)NC2COC2)Cc2ccccc2N(C)CC1C c1(C(N2CCC(CNC(CSC)=O)C2)=O)ccnnc1C Cc1ccc(C(=O)NC2CC(C)CN(C(C3CCOC3)=O)C2)c(N)c1C C1(OC)(CNC(C2CCN2S(C)(=O)=O)=O)CCN(C(=O)C(F)(F)C2CC2)C1 c1(C2C(C=O)C2)cc(F)c(F)c(F)c1.C1(NC(=O)C2CC2)(CF)CCC1 CC(=NO)C1CC(C(=O)N(CC(C)NC(c2ccsc2)=O)C)C1(C)C C1(C(=O)NC(C)C(=O)NCC23CC(F)(C2)C3)CC2OC1C1CC21 C1(CNC(C(c2cncnc2)C)=O)CC2(CC2)CN1C(c1cscn1)=O C1(CC)CN(C(=O)CC2(CO)CC2)CCC1NC(=O)CC1(O)CCC1 Cn1nc(C(F)(F)F)cc1C1(C(=O)NCCNS(N)(=O)=O)CC1 CCC(CC)C(C(=O)NCC12CC(NC(=O)C(CC)SC)(CO1)C2)OC c1(C(=O)OC)cc(C(N2CCCC2CCNC(=O)C(C)SC(C)C)=O)ns1 C1(NC(c2c(C(C)C)csc2)=O)CC2(CCN(C(=O)CC3(C)CC3)C2)C1 Fc1cccc2nc(SCc3ccc(Oc4ccccc4Cl)cc3)[nH]c12 N1(C(c2cc(C3CC3)no2)C(=O)NCC2CCCO2)CC(O)C2(CCOCC2)C1 C1(NC(C2CCC(CC)O2)=O)COC2(C1)CN(C(c1ccc(C(C)=O)cc1)=O)C2 c1(C(N(C)CCNc2ccc(Cl)cc2)=O)c[nH]c(=O)c2ccncc12 C(CCC(C(=O)NCCC1CC(C)(C)C1)NC(c1c[nH][nH]c1=N)=O)OC C1(C(=O)NCC(C)(C)NC(C=CC(C)(C)SC)=O)CC2(CCCCC2)CO1 C1(CNC(C2CCCCC2O)=O)CCCC(NC(=O)C(c2cccnc2)O)C1 c1(C(N2CCC(C)(NC(=O)C=C3CCSCC3)CC2)=O)csc2ccncc12 C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)CCNC(=O)CO)CC1 N1(C(C(CC=C)c2ccccc2)=O)CCN(C(=O)C(C)OC)CC2(C)CCCC12 CCCCCC(F)C(=O)N1CCCC1C1CCCN(C(c2cc(C)oc2C)=O)C1 c1(C(=O)NCC(CNC(C2(F)CCCC2)=O)OC)cc2c(C)cccn2n1 C1(OC)(CNC(C23CC2CCN3C(c2c[nH]nc2C(C)C)=O)=O)CCC(C)C1 C1(NC(C2CCC(C)(C)O2)=O)CC2CC(NC(c3ccc(F)cn3)=O)C2C1 CS(=O)C1CN(C(=O)CC2CCN(C(=O)C=CC(C)(C)C)CC2)C1 c1(-c2cn(CCCN(S(C)(=O)=O)CCC)nn2)ccc(F)c(C(C)=O)c1 N1(C(C(C2CCOC2)OC)=O)CCCC(NC(C2CN3CCN2CC3)=O)C1C c1(C(C)OCC)nc(C)c(C(=O)NC2CCCC(NC(c3cc(C)ns3)=O)C2)s1 CC1=C(C(=O)NC2CCCC2C(=O)NCC2CCC(=O)N2)CCC1 C(CC)(CCC(F)(F)F)(c1n(CCCC)nnn1)NC(c1ccc(OC)cc1)C C1(C)(CNC(=O)OC(C)(C)C)CCC(C(=O)Nc2nccc(-c3ccccc3)n2)C1 C12CN(CC13CC3)C2=O.CC(C)(CF)C(=O)NCCCC1C=NNC1=O N1(C(C(=Cc2ccncc2)C)=O)CCC(N=c2[nH]ccc(C#N)c2[N+](=O)[O-])CC1 N1(C(C#CC(=O)N(C)C)=O)CCC(NC(=O)CCSC(F)(F)F)C(F)C1 N1(C(c2c(C)csn2)=O)CCC(O)C(N(C)C(C2CC(=O)N(C)C2)=O)C1 c1(C(=O)NCC2CC(NC(c3cn(CCOC)nn3)=O)C2)nc(C)n(CC)c1C C1(C(=O)N(C(CC)C(=O)N2CCC(c3nn[nH]n3)C2)CCCO)COC(=O)N1C c1(C(C)C)ncc(Br)c(C(=O)NCC2COCCN2C(C2C=CCCC2)=O)n1 N1(C(C(C)(C)C2CCCCO2)=O)CCCC(CNC(=O)CN2CCOC2=O)C1 Cc1cc(C)c(CNC(C2(C(C)C)CCN(C(C3CN(C(N)=O)C3)=O)C2)=O)cn1 c1(C(=O)NC2CCN(C(C3(C4CC4)CCCO3)=O)CC2O)cccc2c1OCO2 C(=O)(C(CO)NC(C1CC(N(C)C)C1)=O)N(CCN(C)C)C C1(CNC(C2CCSCC2)=O)CC2CCC(C1)N2C(=O)CC1CCCNC1=O c1(C(N(C2CCC(NC(CC=CCC)=O)C2)C)=O)ccc(C(=O)NC)c(F)c1 c1(CN(C)C(C2(N(C)C)CC2)=O)ccc(CNC(c2nscc2Br)=O)cc1 c1(C(=O)NCC2C(NC(C(C(C)(C)C)O)=O)CC2)ccc2c(O)nc(S)nc2c1 N1(C(c2cccc(OC(C)C)c2)=O)CCC(CNC(=O)CC(C)N(C)C)C1(C)C C1(COCCOCCOC)CC(NCC(=O)OS(C)(=O)=O)C1 c1(CC(N2CCC(NC(c3sccc3C3CC3)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 C1(NC(C2CCC2C(F)(F)F)=O)(CO)CCCN(C(=O)Cn2cncn2)C1 Cc1ccc(Br)cc1CC(=O)NC1(CNC(=O)C(F)=CC2CC2)CCOC1 C1(C(=O)C)(C(=O)OC)CCCC1.C1CCCN(C)C(=O)C(C)NC(=O)N1.C1(N)CC1 C(CC(C(C)C)NC(C1(C2CC2)CCCO1)=O)N(C(c1cc(C)sc1)=O)C c1(OCCCC(=O)NC(C2OCCN(C(C(C)OC)=O)C2)C)ccc(F)c(F)c1 C1(C(N(CCCN(C)C)CCC)=O)CCCCN(C(=O)C(COC)OC(C)=O)C1 N1(C(CC(=C)C)=O)CC2CC2(NC(c2c(C)noc2N)=O)C1 C1(NC(C2CCC(CCCC)CC2)=O)CCN(Cc2ccc(O)cc2)CC1F c1(C(=O)NCC2COCCO2)cnc2c(c1)CNC2=O CCCCS(=O)(=O)CC(=O)NC1CCOCC1NC(=O)Cc1sc(O)nc1O C1(C)(C(=O)NC(CC(=C)C)C(=O)NCC)CN(C(C2(N(C)C)CC2)=O)C(C)(C)C1 C(=O)(C(C)CC(=O)NCCN(C(c1ccc(O)cc1)=O)C1CC1)OC c1(NC(C2CCCN(Cc3cc[nH]n3)C2)=O)c(O)cccc1F C1(CNC(c2c(C(C)NC(c3ccn(CCF)n3)=O)n[nH]c2)=O)CCN(C)CC1 N1(C(C(F)=CC)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(n2ccnn2)C1 C1(C(=O)NC(C)Cn2cncn2)CN(C(C2(CO)CCCC2)=O)CC12CCC2 N1(C(C2(S(C)(=O)=O)CC2)=O)CCCC(NC(=O)C(=Cc2cccc(F)c2)F)CC1 c1(CCC(N2C3CC(NC(CCOCCN(C)C)=O)(C3)C2)=O)ccc(N)c(F)c1 C=C=CC(C)C(=O)N(CCNC(=O)CCCCNC(=O)CCCC#N)CC C(=O)(CCCC(C)(C)NC(c1cccnc1O)=O)NC(C)CCN(C)C c1(CN(c2ccccc2)CN2CC(C)C2(C)C)csc2nnsc12 C1(CC(=O)N(CC(N2CCC(OCC=C)C2)=O)CC(C)C)CCCOCC1 C(=O)(C(F)(F)C(F)F)N(C)CC1(O)CCN(C(CS(=O)(=O)N(CC)CC)=O)C1 c1(CC(CNc2c(C(CC)=O)cccc2)N(C)C)cccc(F)c1F N1(C(CC(CC)O)=O)CCOC2(CCN(C(c3cc4c([nH]3)CCC4)=O)CC2)C1 c1(C(N(C)CC2(O)CCCN(C(C(CCSC)O)=O)C2)=O)cccc2c1OCC2 N1(C(C(C)(C)O)=O)CCC2(CC1)CN(S(=O)(=O)CC1CC1)CCO2 Nc1c(C(=O)NCC2(NC(=O)CC3CCC(O)C3)CCOCC2)cc(F)cc1F c1(SC)ncc(C(N2CCC(F)(CF)C2)C(=O)Nc2ccccc2)n1C c1(OC)ccc(CC(C)C(=O)NC2CCC2NC(=O)CN2CC3CC3C2)cc1 Cc1csc2ncnc(NC3CCC3C(C)C)c12 c1(NC2CC3CN(C(C=CC4C(=O)C4(Cl)Cl)=O)CC32)ncc2scc(Br)c2n1 c1(C(N)=O)coc(C(=O)NC23CC(C(=O)NCCCN4CCCCC4)(C2)C3)c1 c1(NC(c2cncc(-c3ccc(SC)cc3C)n2)=O)ccc2nnc(C)n2c1 c1(C(N2CCCC(N(C(C(C=C)(C)O)=O)C)CC2)=O)[nH]c2c(c1C)C(=O)CCC2 Cc1cccc2c(C(=O)NCC3CC3CNC(C3(N(C)C)CCCCC3)=O)coc12 N1(C(CSCCCC)=O)CCC(CO)(CNC(C2(O)CCCCCC2)=O)CC1 C1(NC(C2CC(=C)C2)=O)(CO)CCN(C(C2CCSC2)=O)C1 CC1C(OC(=O)CCc2nc(Br)cs2)CC(=O)N1C c1(C(N(C(CCNC(Cn2c(C)cc(C)n2)=O)C)C2CC2)=O)c(F)cccc1Cl c1(CNC(COCCC)=O)nc(C)c(C(=O)NCc2ccn(C(C)C)n2)o1 C1(C)(C(=O)NCC2OCC(CNC(C=CC(C)C)=O)C2)CCSCC1 C(CC(F)F)(C(=O)NCCc1cn(CC)cn1)N(C(c1c(CC)n[nH]c1)=O)C C1(NC(CN(CC)CC2CC2)=O)(CC)CCN(C(=O)C(C)CC2CC2)CC1 c1(C(=O)NC2(C3N(C(C(C)OC(C)C)=O)CCCC3)CC2)ccc2n[nH]cc2c1 c1(C(=O)NC2CN(C(c3scc(C)c3)=O)CC2C)ccc2ncn(C)c2c1 c1(CNC(C2CCN(C(CN3CCC(OC)C3)=O)C2)=O)cc2cccc(C)c2[nH]1 C1(CCOC)(NC(=O)CCCC(C)O)CCN(C(c2ccncc2SC)=O)CC1 C1(C(=O)OC)CC(COC)CN(C(N2CC3CC3C2)=O)C1 C12(C(=O)NC(CC)(C)CNC(C3C4CC4C4CC34)=O)CC3CC1C2C3O N1(CC2(O)CC(C(=O)NCC3(NC(C4(C)CC4)=O)CCOC3)C2)CCCS1(=O)=O c1(C(=O)NCC(C)(C)NC(CC(COC)C)=O)cccc2c[nH]nc12 N1(C(=O)OC(C)(C)C)CCOC(CCOC(c2sc(Br)cc2Cl)=O)C1 Cc1nc2c(o1)CCCC2CC(=O)N1CC2CC2(NC(=O)CC=C(Cl)Cl)C1 C(CCCC(=O)NC(C(=O)N1CC(c2cccs2)C1)c1ccco1)N(C)C Cc1ccc(C(N2CCC(C)(C)C2CNC(C2CCCCO2)=O)=O)nc1O C1(C(N(CCCNC(c2[nH]cnc2C(C)(C)C)=O)C)=O)CC2(CCC2)CO1 C12(C(N3C(CN(C(C4C(C)OCC4)=O)C)CCC3)=O)CCCC1C2(F)F C1(CC(N2CC(CNC(CCCCC#N)=O)OCC2)=O)Cc2ccccc2C1=O C1(C(=O)OCC)CN(C(=O)OC(C)(C)C)CC2(CCC2)C1.c12ccccc1CO2 CC(CCCCNC(=O)C(=Cc1cccnc1)F)NC(=O)CC1CCCO1 C12(CNC(CN(C3CC3)CC)=O)CCCC1CCN2C(=O)C=Cc1ccnn1C N1(C(C(C(C)C)OCC)=O)CCC(NC(c2ccc(Cl)cc2)=O)CC(C)(C)C1 C1(NC(C(C)Sc2ccc(C)cc2)=O)CCN(C(=O)COC2CCC2)CC1CO c1(C(=O)NC2CN(C(Cn3c(C)cc(C)n3)=O)C(C)C2)ccc(C2CC2)c(C)c1 c1(CC(=O)NC2CC(C)(CNC(c3nc(C)sc3)=O)C2)cnccc1C C1(O)(C(=O)NCC(C)CNC(=O)CCOC2CCC2)CCSCC1 c12cccc(c1)CN2.c1(CCNC(=O)NCCSCCCC)ccc(OC)cn1 c1(C(=O)NCCCN(C(CC2CC(C)C2)=O)C(C)C)ccc(F)cc1F C(C(F)(C(=O)NC1CN(CC)C1)C(C)C)NC(c1c(CC)cc[nH]1)=O Cc1cnn(C)c1C(=O)NCC1(O)CC(NC(C2CCN(C)C2)=O)C1 N1(C(c2ccc(SCC)nc2)=O)C2CCC1CC(NC(C1CCCC1C)=O)C2 c1(CCC)ccc(C(=O)NCCN(C(C)C2CC2)CC)o1 C1(NC(CC2(C#N)CC2)=O)CN(C(c2cncc(Cl)c2)=O)C2(CCCC2)C1 CC(C)(C)C(CNC(c1cnn(C(C)(C)C)c1Br)=O)NC(C1CC12CCC2)=O c1(C(=O)NCCC2CC3CCC(C2)N3)nc2ccccn2c1Br CC1CCC(NC(=O)CC(C)(C)C2CC2)CN1C(=O)CC1CC12CC2 N1(C(C(CSC)OC)=O)CCN(C(=O)Cc2ccc(C)nc2)C(CC(F)F)C1 CCC(CC)C(=O)N(C1CC(C(=O)NCC2CCCC(COC)C2)C1)C Cc1ccc(C)c(CCCC(=O)N2CC(C)(NC(C3CC3c3cccs3)=O)C2)c1 C(=O)(CCCCCF)N1CCC(F)(CNC(=O)CCc2ccccc2)C1 C1(C(N(CC=C)CC)=O)CCCC1CC.C1(C(=O)NC(C)C(=O)OC)CCCC1 C(=O)(C(C(C)C)NC=O)NC(C(=O)N(CCCN(C)C)CCC)C1CC1 CC1CCCCC1(CNC(=O)CCC(N)=O)NC(=O)C(=C1CCCCC1)F N1(C(c2ccc(SC)o2)=O)C2CCC1(CNC(C1(C)CCNC(=O)C1)=O)CC2 n1(CC)nc2c(c1C(=O)NC1CN(C(C3(C(N)=O)CC3)=O)CCC1F)CCCC2 N1(C(c2cc(CCCCC)[nH]n2)=O)CCOCC(NC(=O)CSc2cn[nH]c2)C1 c1(C(N2CC3C(NC(Cc4cnn(C)n4)=O)C3C2)=O)c[nH]c2cccnc2c1=O c1(C(N2CCC(N(C(=O)COc3ccn(C)n3)C)C2)=O)cnc2cccnn12 c12cc(C)n(c1C)c(=O)[nH]2.c1(NC(CCSCC(=O)OC)=O)nccc(C)n1 Cc1csc(=NCC(=O)NC2(C)CN(C(c3cnn(CC(F)F)c3C)=O)C2)[nH]1 C1(NC(C2(CCCC)CCC2)=O)(COC)CCN(C(c2ccncn2)=O)C1 C(=O)(CC(C)(C)C)NCC1C(NC(C(CC2CC2)OC)=O)CC1 C12(C(=O)NCCCCNC(=O)CSCCCc3ccccc3)CCC(CC1)OC2 C(=O)(C(C)(C)C#C)N(CCC(=O)NCC1CC1)CC#C N1(C(C2CC=CC2)=O)CCC(CC2COCCN2C(C2CC=CCC2)=O)CC1 c1(C(N2CCC(N(C(C3(CC=C)CC3)=O)C)C2)=O)ccc2ncccn12 N1(C(C(C(=O)OC)C)=O)CCCC12CCN(C(c1nccnc1C)=O)C2 N1(C(CC(CC)OC)=O)CC2CCN(C(=O)COC(F)(F)F)C2C1C O=C(C#CC1CC1)N1CC=CC(C(=O)NCCC2CC(F)C2)C1 CCCCC(C(=O)NC1(CCOC)CCC1)NC(=O)CC1(N(C)C)CC1 CS(=O)(=O)c1ccccc1CC(=O)NCC1C2CC1N(C(C1(F)CCOC1)=O)C2 c1(C(N2CCCC(CCC(=O)NC3CC3C3CCC3)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(OC)ccc2cc(C(=O)NCCN(C(C3CC4CC4C3)=O)C3CC3)ncc2c1 C=CCCCCC(C(=O)NCc1cccc(OC)c1)N1CCOC(C2CCC2)C1 C(=O)(CS(=O)(=O)CC(C)C)NC1C(NC(c2c(C)oc(Cl)n2)=O)COCC1 N1(C(c2n(C)nc(Br)c2)=O)CC2CCN(C(C3COC3)=O)CC2C1 CC1(CNC(=O)CCF)CCCN(C(=O)C(c2ccc(F)cc2)C2CC2)C1 C1(CNC(c2c(C)cno2)=O)CN(C(C2CC3CC(=O)C2O3)=O)CC1(F)F C#Cc1cccc(C(=O)NC(C(=O)NCC2NC(=O)NC2=O)c2ccoc2)c1C C1(CC(=O)N(CCn2cc(-c3cccnc3F)nn2)CCl)CCc2sccc2C1=O C(=O)(C1=Cc2ccccc2OC1)NCC(CNC(=O)CO)OC n1(CCC(=O)N(CC(C)C)C(C)(C)C)cc(CCN(C(=O)C(O)C2CC2)C)nn1 c1(CC(N2CCCCC2CNCC2CC2)=O)cccc(Cl)c1F.C1(C2CC2)CC1 c1(CC)ccc(C(=O)NC2(CNC(=O)C(C)=CC3CC3)CCCC2)o1 N1(C(C2(C#C)CN(C(c3cnn(CCF)c3)=O)C2)=O)CCn2ccnc2C1C C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CCN(C(c2c[nH]c(Br)c2)=O)CC(O)C1 C1(CNC(=O)CCN2CCOCC2)CCC2(CC1)CCN(C(=O)C1CC1)CC2 CC1CCCC1C(=O)N(C)CCOCCCN(C(=O)CSC1CCCC1)C N1(C(c2cc(C)c(C)o2)=O)CC2CN(C(=O)C(C)c3cc[nH]n3)CC2(C)C1 c1(C(=O)NCC2N(C(CCSCC(C)C)=O)CC2)cncc2ccccc12 C(=O)(C(CC(C)C)n1ccnc1)NC(CCCC)CF c1(C(N(C2CCCC(OC)C2)C)=O)cc([N+](=O)[O-])cc2ccccc12 C(=O)(C(C(C)C(C)(C)C)N1CCOC(c2noc(C(C)C)n2)C1)NCC C=CC1(CC(=O)NC2(COC)CN(C(c3cnc(C4CCCO4)s3)=O)C2)CCC1 c1(C(N2CC(NC(C(C)=C(C)C)=O)C(C(F)F)C2)=O)ccc(Cl)c(F)c1 C(=O)(C(F)C(C)(F)F)N(CCC(=O)NC1CC12CC2(F)F)CC#C c1(C2(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)CC2)cccc(C#N)c1 c1(C(C(=O)N(C)C)C(CC)OC2CN(C(=O)OC(C)(C)C)C2)cccc(C)c1Br c1(C(=O)NC(CC)CNC(C2(C)COC2)=O)ccnnc1O CC1CCN(C(=O)CCNC(C2(C3CC3)CC2)=O)CC1CCOC1CCOCC1 C12(C(=O)NC(CC)CNC(c3ccc(COC)s3)=O)CC3CC(C1)CC(C)(C3)C2 C1(NC(c2ccc(C(C)C)s2)=O)C2CC1CN(C(=O)C(C1CCOCC1)O)C2 Cc1c(C(C)NC(COC(C)(C)C)(CF)c2nnnn2C)sc2cncn12 c1(CN(CCO)CC2N(C(Cc3ccn(CC)n3)=O)CCC2)ccnc(F)c1 Cc1nc2ncccn2c1C(=O)N(C1CC2CC1CN2)c1cc(Cl)n[nH]1 C(=O)(C(O)CC(C)C)NCC1(O)CCN(C(c2ncn(CC)c2)=O)C1 O=S(=O)(c1ccc(Br)cc1NC(CF)CF)NCCN1CCC2(CC1)CC2 c1(NC(C2CN(C(C34C=CC(CC3)C4)=O)CC2n2cccn2)=O)ccc(F)nc1 C1(CNC(CCC)=O)CN(C(c2nc(Br)c[nH]2)=O)CC12CCC2 N1(C(c2c(C)cc(CO)o2)=O)CC(CNC(c2coc(CO)c2)=O)CCC1C c1(C(N(C(C)CNC(C2(n3nccn3)CC2)=O)C)=O)ccc2c(c1)OC(C)(C)O2 c1(N(C)C)ccc(C(=O)N(C2CCN(C(c3ncccn3)=O)CC2)CCO)nc1 CC1CCN(C(=O)CCc2cccnc2)C(CNC(=O)CCc2cnc[nH]2)C1 c1(CC2C(=O)N2)ccc(C(F)F)cc1F.CCCC(O)CNC(=O)COC(C)C C1(CCC(=O)NCCOC2CN(C(c3csc(-c4cccs4)n3)=O)C2)CCCOC1 C1(C(=O)NC23CC(CNC(c4nc(OCC)oc4)=O)(OC2)C3)C(F)(F)C12CCC2 c1(CNC(c2ccc(Oc3ccccc3)c(Cl)c2)=O)ccc2c(Br)cccc2c1 c1(C(N2CC=CCC2CC)C(=O)NCCOCC)ccc([Si](C)(C)C)s1 C1(C)(CN(C)C(C2CC2CNC(c2csc(Cl)c2)=O)=O)CCCC1 C(=O)(CC1=CCN(C(=O)CO)CC1)C(CN1CC(C)C1)=O.C(CSCO)N S(=O)(=O)(c1cnc(NC(c2ccc(C)s2)C)c(Cl)c1)NCC(CC)(C)COC C#CCCN=C(NCC1CCN(C)C1)NCCc1cn(C)c2ccccc12 C1(CNC(c2cccnc2)=O)(OC)CN(C(c2c[nH]nc2-c2cccnc2)=O)C1 CC(CC(F)F)C(=O)N1CCC(O)(CCNC(=O)COc2ccc(F)c(F)c2)C1 c1(COC)nc(CNC(=O)C(C2CCOC2)NC(C2CC(C)(C)C2)=O)no1 c1(C(N2C(C(=O)NCC#C)CCC2)C(=O)NCC2CC2)cnn(CC)c1C C1(C(N2CC(COC)(CNC(=O)C=CC(C)C)C2)=O)CCc2ncc(C)n2C1 N1(C(C(CCC)Cl)=O)CCC2(CC(C(N3Cc4ccccc4C3=O)=O)CO2)C1 Cc1nn(C)c(C)c1C(N1CCOC(C(N2CCC(O)(C(N)=O)C2)=O)C1)=O n1(CC)nc(C2CC2)cc1C(N1CC2CC1C2NC(=O)CC1COC(=O)C1)=O C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(c1ccnc(C(=O)OC)n1)C2 c1(C(=O)NCCN(C(c2ccoc2)=O)CC)ccc(OC(C)C)c(C#N)c1 C(=O)(C(N=[N+]=[N-])C(C)C)N1CC(OCC(=O)NCC2N(CCOC)CCC2)C1 C1(NC(C(CC)Oc2ccc(Cl)cc2)=O)CCN(C(c2csc(C)n2)=O)CC1O N1(C(C2(COC)CC=CC2)=O)CCC2CN(C(C3CCc4ccnn4C3)=O)C2C1 c1(NC(c2cccc(C3(COC)CCCCC3)c2)=O)cc(=NCCCSC)[nH]cn1 C=CC1(NC(C2(CNC(=O)CC(C)OC)CCC2)=O)CCOCC1 C1(NC(C(CNC(c2c(C)ccs2)=O)CC2CC2)=O)CC2(CCC2)C1O C1(CNC(C(=O)NCC2(C3CC3)CCCO2)=O)CCN(c2ccnc(CO)n2)CC1 c1(NC(N(CC(C)(C)C(F)(F)F)C)=O)ccc(C#N)c(Cl)c1 C12(NC(C(CSC)O)=O)CC(CNC(=O)Cc3ccc(C)c(C)c3)(C1)OC2C C=CCCCCC(=O)N1CC(CNC(C2CC2c2cccs2)=O)C(O)C1 C(CC(CO)NC(=O)Cc1csc(-c2ccsc2)n1)=CC N1(C(c2ccc(SC)s2)C(=O)NCC)CCC(F)(F)CC1C c1(CN2C(C(=O)Nc3ccc(C)nc3)CC(F)C2)ccc(C(F)(F)F)nc1Cl c1(C(N2CCC(CNC(C(C)CF)=O)C2)=O)cc(Br)ccc1O N#Cc1ccccc1CNC(Cc1ccoc1)CO c1(C(N2CC(NC(CCc3n(C)ccn3)=O)C(CO)C2)=O)n[nH]cc1[N+](=O)[O-] C1(CNC(C(Br)=C(C)C)=O)CC2COCC2N1C(c1coc(C(N)=O)c1)=O C1(C(=O)NCC2N(C(C3(C)CC(=C)C3)=O)CC2)CCC(c2ccccc2)CC1 C(=O)(C1Cc2ccccc21)N1C2(CN(C(C3(C)CCCCO3)=O)C2)CC1 C1(C(=O)NCCCCNC(CC(=O)N(CC#C)C)=O)C=CC=CC=C1 CCC(C(=O)N1CC(CC(=O)NC(C)(CC)CO)(OC)C1)C(C)C CC(C)C(C)C(CNC(=O)CCc1ccc(F)cc1)NC(=O)C(F)=CCCF Cc1c(C(=O)N(CCCNC(C2CC23CC3)=O)C2CC2)cccc1[N+](=O)[O-] Cc1nc(C2(NC(=O)NC3CC3OC(C)(C)C)CC2)no1 c1(C(N(C)Cc2nnc(C)o2)=O)nc(CNC(=O)CCc2nccn2C)oc1C Cn1ccnc1CCC(=O)NCCN1CCC(NC(c2c[nH]nc2C(F)F)=O)C1 N1(C(COCCC=C)=O)CCOC(CCCNC(=O)CC2CC=CCC2)C1 Nc1ccc(C(=O)NCC2CN(C(S(=O)(=O)C3CC3)=O)C2)cc1[N+](=O)[O-] c1(CC(N2CCN(C(=O)COC(F)F)C(CC(F)F)C2)=O)ccc(F)c(F)c1 c1(C(=O)NCCOCCN(C(C2(C(=O)OCC)CCC2)=O)C)ccc(C)c(F)c1F C1(C(C)C)CN(C(c2ccc(N)cn2)=O)CCCN1C(c1cc[n+]([O-])cc1)=O C1(C)(C(N2C(CNC(c3cc(C)no3)=O)CCC2)=O)CC(C#N)C1 c1(C(N2CC3C(C(N4CC(OCC)C4)=O)C3C2)=O)ccc2c(c1)CC2 C(=O)(C(O)C(C)(C)CC)NCc1cccc(NC(c2nncc(CCC)c2)=O)c1 c1(C(=O)NCCN(CCC)C(C2(c3ccc(C)o3)CC2)=O)ccc(F)cc1Br C1(NC(=O)Cc2cncc(F)c2)CN(C(=O)CN2CCSCC2)CC1C(F)F CC1CN2CCN1C(C(N1CC3OCC(NC(C4CCC(=O)NC4)=O)C3C1)=O)C2 CC(C)CC(C)(O)CNC(C1CCCC(NC(c2cc(Cl)n(C)n2)=O)C1)=O N1(C(CCn2cc(C3(S(=O)(=O)N(C)C)CC3)nn2)=O)C2CCC1CC(CC(F)F)C2 Cc1cnc(NC2CCN(C(c3nn[nH]c3C(F)(F)F)=O)CC2C)nc1C c1(CCC(=O)NCC2CCN2C(=O)C=CC2CCC2)ccc(Cl)nc1 Cc1ccccc1CNC1CCC(CNC(c2ccccc2Br)=O)CC1 c1(C(N2CCOC3CCCCN23)C(=O)NCCCOC)cc(C)c2occc2c1 CC1CN(C(=O)C=C2CCOCC2)CC1CCNC(c1cnc(C2CC2)nc1)=O c1(NC)ccc(-c2cnc(OCC3CC3)c(C(N3CCOC(C)C3)=O)c2)cc1F C#Cc1cccc(C(=O)NC(C)(CSC)C(=O)NCCCC(=O)OC)c1 Cc1nn2cc(CC(=O)NCC3CC(NC(=O)C(c4ccccn4)C)C3)nc2s1 C(=O)(CC(O)C(C)(C)C)NCCN(C(C)C)C(C1CCc2nc[nH]c2C1)=O N1(Cc2ccc(C)cc2)CCC(NC(c2ccc(C(C)C)s2)=O)CC1C c1(C(=O)NC(C2CC2(Cl)Cl)C)ccc(OCC2CC2)c(F)c1 Cc1sc(C(=O)NCC(O)CN(C(=O)Cc2ccc(O)nc2)C)nc1Br CC(CC(C)(C)C)NCCc1ccc(Cl)cc1 n1(CCCC)nc(C(=O)NC23CCC2CN(C(C24CCC2CC4)=O)C3)ccc1=O c1(N(CC(C)NC(c2ccc(N3CCCC3=O)cc2)=O)C)snc(Cl)c1C#N N(C1CCc2cccc(Cl)c21)C(=O)Nc1ccc(SCc2ccc(C)cc2)cc1 CC1(C)C=C(C(=O)NC2(C)CCCCC2C(N2CCOC(C3CC3)CC2)=O)C1 N1(C(c2cn(CC)nc2C2CC2)=O)CCC(NC(=O)Cn2cncc2C)C12CC2 c1(NCC(CC)(CC)NC(C2CC3CCC2O3)=O)cc(C)nc2c(C)cnn12 c1(OC)cnc(Cl)[nH]c1=NC(=O)C1(CNCc2ccc(C)cc2OC)CC1 C1(F)(C(N(CC(CC)(F)F)C)=O)CCN(C(C2CC23CC3(F)F)=O)CC1 N1(Cc2c(C)ccc(OC)c2)CC2CCN(C(=O)C(=O)c3ccco3)CC2C1 c1(NC(C)=O)nc(C(=O)NCC(C)NC(=O)Cc2cnn(C(C)(C)C)c2)cs1 CC(CCCCO)NC(c1ccc(CNC(C2CCC2(F)F)=O)cn1)=O C(=O)(CC(O)CNC(=O)CC(C)NC(=O)CCc1cccn1C)OC C1(C(=O)NC(CNC(C(C)CS(C)(=O)=O)=O)C2CC2)CCC2C(CC1)C2(F)F n1(CC(=O)NC(CC(C)C)CNC(=O)Cc2ccns2)nc(Cl)ccc1=O C1(CC)(NC(c2ccc(=O)n(C)c2)=O)CCCN(C(=O)Cc2cnc(C)s2)C1 c1(NC(C(c2ccc(C)cc2)=O)=O)ccc(NCc2ccc(Cl)c(Br)c2)cc1F O=C(CC(C(F)F)N1CCOCC1)NC1CCCN(CC2CC2)C1 O=C(C1CCCc2cncn21)NC1CCC(NC(c2cnc3[nH]cnc3c2)=O)C1 O=C(CCCCCNC(C1(O)CCSC1)=O)NCc1ccncc1Cl N1(C(CC2CC(OC)C2)=O)CCC(CNC(=O)C(C)CN(C)C)C(O)C1 c1(CN2CCC(C(=O)NCCCSC(F)F)C2)ccc2ccoc2c1 C(C(C)(C)CC(=O)NCC(CC1CCCC1)C(=O)NCC(C)(O)CSC)OC C(C(F)(F)C(C)(C)O)NC(C(C)NC(C(C)c1cccs1)=O)=O c1(C(=O)NCC2(NC(CN(C)CC)=O)CCOC2)ccn(CC(F)(F)F)c(=O)c1 CN1CCCC(C(C)(C)C(=O)N2CC(CNC(C3(C#N)CCOC3)=O)C2)C1 N1(C(C2(C=C)CCOCC2)=O)CCC2CC(C1)CN(C(=O)Cn1cnnn1)C2 N1(C(COC(C)=O)=O)CC(NC(=O)C(C)C2CCC2)Cc2ccccc21 C1(CNC(C=Cc2cn(C)nc2)=O)CCCCN(C(C2CN3CCC2CC3)=O)C1 Cc1nc2c(N3CC4(CN(C(=O)C(C)(C)CCl)C4)C3)ncnc2[nH]1 c1(C(=O)NCCC2CCN(C(C3(O)COC3)=O)CC2)cncc2c(Cl)cccc12 Cc1nn(C)c(C(N2CCC(CNC(c3ccc(Br)c(F)c3)=O)C2)=O)c1F CC1CCN(C(C23CCCC2CCC3)=O)CC1NC(=O)CC1CCCSC1 Cc1[nH]nc(C(N2C3CCC2CC3)=O)c1O.C(CC(=O)O)NC(C)C c1(NC(C(NC(=NC)NCCCC(=O)OC)C)OC)ccc(N2CCOCC2)cc1 N1(C(C23N(C(CC(=O)N(C)C)=O)CC(C2)C3)=O)CC2CC1CN2C(N)=O CC1CC(C)(C)CCC1NC(=O)C(C)(C)CCNC(=O)C=Cc1ccc[nH]1 N1(Cc2cnc(-c3cc(C)c(F)cc3)s2)CCC2(CC1)OCCO2 C=CCCN=C(NCc1ccc(C)s1)NCC1CCOC1c1cnn(C)c1 CC1CCCN(C(C2CCCCCCC2)=O)C1CNC(C1CCC1)=O N1(C(C(=CC2(C)COC2)C)=O)CCC(C(N2CCC(C(C)C)C2)=O)C1(C)C C1(CN(C(C)C)C(C2COCCO2)=O)CN(Cc2nnn(C)n2)CCO1 CC(CC(=O)NCCCN(C)C(C1CC(C)(C)OC1(C)C)=O)C(C)(C)C CC(c1ccccc1Cl)=CC(=O)NC1CN(C(C2(NC3CC3)CCC2)=O)C1 c1(C(=O)NC2CC(N(C(=O)CCc3n[nH]c(=N)s3)C)C2)nnc2ccccc2n1 C1(N(C)C)CCCC(C(=O)NC(CNC(=O)C=C2CCN(C)C2)CO)C1 CC1(CNC(C2CCCN2C=O)=O)CCN(C(c2cccc(C#N)c2)=O)CC1 Cc1cc(C(=O)NCc2ccoc2C(N2CCC(OCC(C)C)C2)=O)no1 Cc1nn(C)c(C)c1-c1cn(CC2CN(C(=O)C(F)OC(F)(F)F)C2)nn1 C1(NC(C2(CCNC(CC(C)OC)=O)CC2)=O)CCCC(O)C1O c1(OC)ncc(F)cc1-c1cn(C2CSCCN2C(C2CC(O)C2)=O)nn1 c1(C(N2CC(O)(CCNC(CC(C)SC)=O)C2)=O)cnc(C(F)(F)F)nc1 N1(C(=O)CNC(c2cnco2)=O)CCC2CN(C(c3ccco3)=O)C2C1 c1(C(N2CC(C)C(NC(c3cccs3)=O)C2)=O)cc(Br)c(F)cc1N c1(C(N2CC(CNC(C(C=CC)O)=O)C(O)C2)=O)ccc(C)c(Br)c1N c1(C(=O)NC(C2N(C(C=C(C)C)=O)CCCC2)C)cnc(C2CCC2)nc1O CC(C(=O)NCc1ccc(C(=O)NCCP(C)(C)=O)cc1)C(F)F N1(C(C(C)=O)=O)CC2(CCCN2C(c2cc(F)ccc2-n2nccn2)=O)C1 Cc1cc2c(C(N3CCN(C(=O)CC4CCCO4)C(C(F)F)C3)=O)cccc2o1 CC1(NC(=O)CNC(C2CC(=C3CC3)C2)=O)CCCOC1 C(=O)(CC(C)P(C)(C)=O)NCC(CN(C(C(C(C)C)NC(C)=O)=O)C)(C)C C1(NC(C(CC)C)=O)CC(C2CCN(C(=O)CCCN(C)C)C2)C1 C=CC(CCC)CC(=O)N1CCCC(C(=O)NCCc2ccsc2)C1CC Cc1cc(=O)c(C(=O)NC2CC(=O)CN2C(=O)COC2CCOCC2)c(C)[nH]1 c1(C(=O)NC(C(=O)NCC2CCO2)C2CCOC2)cnn(CCO)c1 c1(CC(=O)NC2CC(F)CN(C(c3cc(OC)ccn3)=O)C2)cc(O)nc(O)n1 CN1CCN(C(=O)C#CC2CC2)C(CNC(c2cn(C)c(=O)n2C)=O)C1 c1(NC(C2CCN(CCCNC(C(CC)O)=O)C2)=O)cc(F)ccc1OC N1(CCNC(=O)CC2CCCC2)CCC(O)(CNc2ncc(Cl)cn2)CC1 C12(NC(CS(=O)(=O)NCC)=O)CCCC1CN(C(=O)CC1CN3CCC1CC3)C2 c1(C(=O)OCC(C(=O)OCC)CCSc2ccccc2)csc2ccccc12 C1(CN(C(=O)CCc2cnccn2)C)CCCN(C(C2COCCO2)=O)C1 c1(C(=O)NC(C)C)cc[nH]c(=NCCNC(=O)C2=COCCC2)n1.C(C)(C)(C)N Cc1[nH]c(C#N)cc1C(=O)NCC1(C(=O)NCC2CCCC(C)O2)CC1 N1(C(CC(CCC)NC(=O)CC2(OCC)CCC2)=O)CCOC2(CCC2)CC1 c1(CN2C(C(N3CC(C(N)=O)OCC3)=O)CCCC2)c(O)ccc2ncccc12 C(=O)(CCC(C)(C)[N+](=O)[O-])OCCCN(C1CCCCCCC1)C c1(C(=O)NCC2C(C(N(C(C)C)CC3CC3)=O)C2(C)C)cc(O)ncc1F C=CCC(C)(CNC(c1conc1C(C)NC(=O)C(C1CC1)SC)=O)CO c1(C(N2CC(n3cc(-c4ccn(C)n4)nn3)C(O)C2)=O)cc2cn[nH]c2cn1 c1(NC(C2N(C(c3c(C)nccc3)=O)CCOC2)=O)cccc(O)c1C C1(NC(c2c[nH]c3nccc-3c2)=O)CN(C(C2CC3CCC3C2)=O)CC12CCC2 c1(C(=O)NC2CC(NC(=O)CCc3ccoc3)C2)c(O)nc(=O)n2c1CCC2 c1(SC)ccc(C(=O)NCC2CC2NC(c2ccncn2)=O)cc1Br C1(C(C)(C)CNC(C2CCCC2F)=O)CCCN1C(C1(C2CCCO2)CC1)=O CCC(C)(COC)C(=O)N1CCC(CN2CCN(C(=O)C(C)CSC)CC2)CC1 c1(C(N(C(CNC(c2nccc(C(C)=O)c2)=O)C)C)=O)ccc(C)c2c1CCC2 N12CCC(C1C)NC(=O)C1(CCC1)C2=O.c1(OCC)cncc(COC)c1 Cc1ccncc1CCNC(C12CC1CN(C(c1ccc(CO)o1)=O)C2)=O c1(CN2CC3CN(C(=O)CC4CC4)CC32)nccc2ccccc12 C1(C(C)C)CN(C(C2CCS(=O)(=O)C2)=O)CCCN1C(=O)C1=NNC(=O)CC1 C1(NC(c2c[nH]cc2Br)=O)CC2(C1)CC(CNC(C1C3CCC(=O)C13)=O)C2 C(=O)(CCCCC(C)C)NCC1(CNC(c2c(C)ccnc2Cl)=O)CCCC1 N=c1nc(-c2cccc(F)c2)nc(N2CC(CNC(C3CCCC34CC4)=O)C2)[nH]1 CCC(C)C(C(=O)N1CCCC1CN(C(=O)CCc1cnc[nH]1)C)OC c1(OC)ccc(Br)c(C(N2CC(NC(c3cncs3)=O)C(F)(F)C2)=O)c1 C1(C(=O)NC2C(NC(c3ccccc3Br)=O)CC2)CCc2nncn2C1 CC1OC(C)C(C(N2CCCC(N(c3cc(Cl)nc(C4(C)CC4)n3)C)C2)=O)C1C C(=O)(C(F)(F)C(O)C(C)C)NC1CC(N(C(C2N(C(C)=O)CCOC2)=O)C)C1 CCC(CC(=O)N1CC(F)CC1Cn1ncc(C(N(C)CC)=O)c1C)C1CC1 N1(C(c2c(C)con2)=O)CCC(NC(c2ccn(CCF)n2)=O)C(O)C1 C1(CC(=O)NC2CC(C(=O)NC3(c4c(C)cno4)CC3)C2)OCCCC1(C)C N1(CC(=O)NCCC(=O)N(CC(C)O)C)C(=O)CCCC1=O C=CCC(C(=O)NC(C(=O)NCCCCCCOC)C(C)(C)O)C(C)C CCCCCC(=O)N(C)CC1COCCN1C(C1CC1(CC)CC)=O c1(NC(=O)NC2CC(C(C)(C)C)C2)cccnc1 CC1(C(N2CCC(c3cccs3)CC2)=O)CCCCCCC1 N1(C(C(c2cccc(C)c2)O)=O)CC(C2CCN(C(c3ccc(=N)[nH]n3)=O)C2)C1 C1(NC(COCCC=C)=O)CN(C(c2ncsc2C2CC2)=O)CC2(CC2)C1 C=C1Cn2c(C(=O)NC3CCCCN(C(=O)C(C)(O)C4CC4)C3)nnc2S1 Cc1cc(C(=O)NC(CNC(=O)C=CC2CC2)C(C)C)n[nH]1 c12cc(on1)CNC2=O.c1(C(=O)NCCNC(=O)OC)cc(C2CC2)[nH]n1 CN1CCC(NC(C2(CNC(c3cc(C4CC4)on3)=O)CCCO2)=O)C1=O CC(CC(=O)NC1(CNC(c2conc2C2CCC2)=O)CCOC1)n1ccnc1 N1(C(c2c(C)scn2)=O)CC(NC(=O)CC2C=CS(=O)(=O)C2)C(C)(C)C1 N1(C(CN(C)C(=O)C2CC2)=O)CC(F)(CNC(=O)C(C)(C)C2CCCCO2)C1 C(=O)(CS(=O)(=O)CCO)N(C1CCN(C(C(F)SC)=O)CC1)CCO N1(C(C(c2cccs2)NC(CCCOCCC)=O)=O)CCC(F)CC1 N1(CC(=O)NC(CCN(C(C(C)NC(C)=O)=O)C)C2CC2)C(=O)C(=O)N(C)C1=O N1(C(c2oc(C)c(CO)c2)=O)CCC(NC(=O)C(C)c2cccs2)C(C)C1 N1(C(=O)NCc2nc(COCC)sc2)CCc2nc[nH]c2C1c1cccnc1CC c1(C(=O)NCC2C(NC(C3(N(C)C)CCCC3)=O)CCC2)cc(F)c(O)c(F)c1 N1(C(COCCN(C)C)=O)CCCC(CNC(=O)CCn2cnnn2)CC1 C1(CNC(C(=Cc2ccco2)C)=O)CC(O)CN1C(=O)C(=O)NCC(F)F c1(C(N2CCC(F)(C(=O)NCCn3cnccc3=O)C2)=O)cccc2occc12 Cc1nc2nccc(N3CCOC(C)(CNC(=O)C(C4CC4)C4CC4)C3)n2n1 C=CCN=C(NCCSC1CCCC1(F)F)NCC(=O)OC N1(C(C(C)SC)=O)CCOC2CCN(C(=O)CCCN(C)N=O)CC12 N1(C(c2nc(C)[nH]n2)=O)CCOC(CNC(C2CCC23CCC3)=O)C1 c1(-c2nnc(C)o2)ccc(Cl)c(SS(=O)(=O)Cc2cccc(F)c2F)c1 c1(OC)cccc2c1OCC(NC(c1nn(-c3ccccc3)c3c1CCCC3)=O)C2 N1(C(CNC(C)=O)=O)C(CC(=O)NCC(O)CC(C)C)C2CCCC12 c1(C(C)NCCC(CCCC)O)ccc2cc[nH]c2c1 c1(C(N2CC(NC(c3cnc(S)[nH]3)=O)C(CO)C2)=O)c(Cl)ccc2c[nH]nc12 N1(C(CCC)=O)CCC(C)(C)C1CC(=O)N(C)Cc1ccccc1OC C1(CNC(c2c(CC)nc[nH]2)=O)CCN(C(c2cc(C(C)=O)cn2C)=O)C(C)C1 C(=O)(C1=NNC(=O)C1)NCc1cn(CCNC(c2cc(C)nn2C)=O)nn1 C1(NC(C(CC)F)=O)CCCC12CN(C(=O)C1=C(C)CCCC1)C2 Cc1cc(C)c(C(N2CCCC(C)(NC(C3CCC(C)(F)CC3)=O)C2)=O)c(S)n1 CC(=O)CCCC(=O)NC1(C(N2CCCC(C)(CO)C2)=O)CC(F)C1 C1(C2C(NC(c3c(CC(=O)OC)ccs3)=O)C2)CCCCN1C(c1cnc[nH]1)=O C1(CC)CC(O)CN1C(c1nc(NC(=O)CCCCCl)cn1C)=O c1(C(C(N2CCC(N(C(C3CC(=C)C3)=O)CCSC)CC2)=O)O)cccc(C)c1F CC(C)(C)CCC(=O)N1CCCC(NC(C2(n3cc(Cl)cn3)CC2)=O)C1 c1(C(CC)C)cccn1CC(=O)N(CC(=O)O)CCOCCOC c1(CN2C(C(=O)Nc3cc(O)ccc3Cl)CC(O)C2)nc2ccccc2[nH]1 C(=O)(CCCC(C)c1ccccc1)NC1(C)CCN(C(COC(C)=O)=O)C1 C12(C(=O)NCCN(C(C(n3ccc(C)n3)C)=O)C)CC3CC(C1)CC(C)(C3)C2 Cc1ccc(NNC(=O)C2CC(=O)N(CC(F)(F)F)C2)cc1C Cc1ccc(S(=O)(=O)NCC(=O)NC(C)CCCCNC(=O)C(F)=C2CC2)cc1 C#Cc1cccc(C(=O)NC(CNC(C2(SC)CCC2)=O)C2CC2)c1F N1(C(C(CCOC)OC)=O)CC(NC(=O)C(CN(C)C)CO)C2(CCC2)C1 C(=O)(CC(C)C(F)(F)F)N1CCCC(CC)C1C(=O)N(C1CCOC(C)C1)C N1(C(c2cnc(OCC)s2)=O)CC2CS(=O)(=O)CC2(NC(=O)C(N)=O)C1 N1(c2cc(NCC3CCCC(=O)N3)nc(C(C)C)n2)CCC2(CCNC2=O)CC1 C=CC1(C(=O)NC(CC)CCOC)CCN(C(c2cc(F)c[nH]2)=O)C1 C1(C(N2C(C)(C(=O)Nc3c(OC)nc(Cl)cn3)CC2)=O)CCc2ccccc2C1 C12(NC(=O)NC(c3nccn3C)C(C)C)CC1CN(C(=O)C1CC1)C2 CCC(O)CC(=O)N1CCC(C2CCCCN2C(=O)Cc2cncn2C)CC1 c1(N(CCC)CCOCc2cc(C)c[nH]2)ccc(-c2nn[nH]n2)cc1 c1(C(N2CCC(C(C)CNC(=O)CC3OCCO3)CC2)=O)cc2ccsc2s1 N1(C(c2[nH]c(=NCC)sc2)=O)CCC2C(CCCN2C(=O)C=C(C)C(F)F)C1 Cn1ccc(CCC(=O)NCC2CCN(C(=O)C(O)C3CCCC3)C2)n1 C(=O)(CC(C)C(F)F)NCCOCC(=O)NCC(CC(=O)OC)O CC(C)C(C)C(=O)N1CC(O)(C(C)NC(c2c(-c3ccccc3)noc2Cl)=O)C1 N1(C(CCC(O)CO)=O)CCC(=CC(N2CCCC2CO)=O)CC1 n1(CC(=O)NC(c2ccccc2)C(=O)NCC(COC)(F)F)cccnc1=O C12(C(=O)NCc3ccc(C)o3)CCC(CC1NC(=O)C(CN(C)C)N(C)C)C2 c1(OC)ncc(C(N2CC(OC)CC2CNC(c2ccnnc2S)=O)=O)cn1 c1(C(N2CC(C(C)NC(=O)C3=CCCS3)C2)=O)c(F)c(F)c(F)c(F)c1F c1(C(N(C(C)C)CC)=O)ccc2c(C)c(C(=O)Nc3ncc(C#N)s3)[nH]c2c1 N1(C(C(CCC)OC)=O)CCCCC12CC(NC(=O)CCN1CCCCC1=O)C2 C#Cc1ccc(C(N2CC(NC(c3ccc(OC)s3)=O)CC2C)=O)c(F)c1 Cc1[nH]c(C#N)cc1C(N1CCCC(CCNC(c2ncc(Cl)nc2Cl)=O)C1)=O CC1c2c(Br)cnn2CCN1Cc1cc2ccc(F)cc2nc1O C1(C(=O)NC2C(C)CN(C(C3CC(CCF)C3)=O)C2)Cc2ccccc2O1 CN1CCN(C(c2cccc(=S)n2O)=O)C(CNC(=O)CC2(C)CC2)C1 c1(Cc2ccc(N(C(C)Cc3cccnc3)C(C)=O)cc2)nc(=N)[nH]c(=N)[nH]1 Cc1cc(Cl)c(C(=O)NCC2CCN2C(=O)Cn2cccc(O)c2=O)cc1F N1(C(c2c(Cl)cc(C)s2)=O)CCC2CN(C(c3nocc3C(C)C)=O)CC12 CC1(C)COCCC1CC(=O)NCCOC1CN(C(=O)CNc2nccs2)C1 C1(NC(C2CCC(=O)O2)=O)CC(F)CN(C(=O)CSC2CCS(=O)(=O)C2)C1 C(=O)(CCC(=O)NCC1(NC(c2ccc(C)nc2)=O)CCC1)NCC C(=O)(C(C)(C)C(C)(F)F)NCC1CC(C)(C)N(C(=O)CC23CC(C2)C3)C1 c1(N(CCNC(C(CC)OC)=O)C(C)C)cc(CSC)ncn1 c1(OC)ccc(CN(C)CC2CCC2(F)F)cc1 c1(OC)ccc(C(=O)NC2(CCNC(=O)CC3CC(C)(C)CO3)CCC2)cn1 C(=O)(C1=NOC(C)C1)NC1CC(CCNC(c2c(C)ncn2O)=O)C1 CC(C(=O)NOCc1ccccc1)N(C)C(C1CCCS1)=O C1(C(=O)NCC(CN(C)C(c2cc(-c3cccnc3)on2)=O)O)(CO)CCCO1 C1(C(=O)N(C)CCN(C(=O)C(c2ccccc2)C2CC2)C)(OC)CCS(=O)(=O)C1 c1(C(N(C(C)CNC(=O)CSS(C)(=O)=O)C)=O)cc(F)c2[nH]nnc2c1 c1(C(N(CCOCCNC(C(n2c(C)ncc2)C)=O)C)=O)cc(N)c(O)c(F)c1 N1(CC(=O)N2C3CC(C3)C2=O)CCOCC1.c1(CC(=O)NC(C)(C)C)cccs1 CC1CC(C(=O)N(C)CCOCCNC(=O)CC2CCN(C)C2)CCC1C C1(NC(CC2C(C)C2)=O)CN(C(C2CCSC2)=O)CC1O C(=O)(CCCCC1CC1)NCC1(C(=O)NCCC(=O)OCC)CCC1 C1(CNC(C(C2CCOC2)OC)=O)CN(C(C2CN(C)CCO2)=O)CC1O CC1(C(=O)NCCN2CCCCC2)CCN(C(=O)C2(C)CC2)C1.N1(CC=O)CC=CC1 N1(Cc2ccc(COCC)o2)CC2(CC2C(N2CCN(C(C)=O)CC2)=O)C1 C1(CNC(CCC2(C)CC2)=O)CC2COCC2N1C(c1cccnc1C(F)F)=O C1(C(=O)NC2CC(N(C(=O)CC3CSC3)C)C2)CC1C1CC(F)(F)C1 c1(NCC(C)C#N)nccc(=NCC2(C3CC3)CCC2)[nH]1 C1(CC(=O)N(CCC)CC)CN(C(=O)CCc2nccs2)CCC1C N1(C(C(CC)C#N)=O)CCC2(CC1)CC(NC(c1ccc3c(c1)CC(=O)N3)=O)C2 N1(C(C2(CC=C)CCCN2C(=O)C(C2CCCCC2)O)=O)C2CCC(C2)C1CO Cc1nn(C)c(C)c1CCC(=O)NC1CC2CC1N(C(=O)Cc1cnc[nH]1)C2 C(C(O)CCNC(c1c[nH]cc1C1CC1)=O)NC(c1cc[nH]n1)=O S(=O)(=O)(c1ccc(NC2CCOC(C(C)C)C2)c(Br)c1)N(CCSC)CC c1(C(=O)NCC2(C(=O)OCC)CC2C(F)(F)F)cc2cccc(Br)c2o1 C1(OCC(=O)OC)CN(N2CCCCN(C)CC2C(=O)OC2CC2)CC1C(F)F c1(CNC(=O)C(c2ccc(Cl)cc2Cl)(F)F)cc(Cl)ccc1F CC1CCCCC1CC(=O)NCCCC(C)(C)NC(=O)CCn1ncn(C)c1=O C1(c2cccc(F)c2)(C(=O)NC(C2(O)CN(C(C3CC3F)=O)C2)C)CCOCC1 c1(C(N(CCNC(C2(CC#C)CCC2)=O)C2CC2)=O)ccc2c(c1)COCO2 c1(OC)cc(C(N2CC3(CC(=O)N3)C2)=O)c(-c2ccccc2)cc1OC N1(C(C(C)=CC2CC2)=O)CC(C(=O)NC2CCOCC2F)C2(CCC2)C1 C(=O)(C1CCCCc2ccccc21)N(C)CC1CCN(C(C2CC=CC2)=O)CC1 C1(NC(c2ccnc(C)n2)=O)COC2(C1)CN(C(c1ccc(C)cc1O)=O)C2 Cc1ncc2n1CCC(C(=O)N(C)CC1CN(C(=O)Cc3cn[nH]c3)CCO1)C2 Cc1cccc2[nH]c(=NCC(C3CCCC3)NC(=O)CCc3cn(C)nn3)oc12 c1(NC2C(CC=C)CCCC2)ncc(C)cc1S(C)(=O)=O N#CC1CCCC(C(=O)NCC2COCC2NC(c2ccon2)=O)C1 Cc1coc(C(=O)NCC2CCCC2C(=O)NOCCO)c1 N1(C(CC2CC(C)C2)=O)CCC(CC(=O)N(CC(C)(C)CO)C)CC1 C12(C(=O)NCC(CC=C)NC(=O)CCCc3ccncc3)CCC(CC1F)C2 N1(C(C(C=C)OC)=O)CCOC(C2CN(C(C3CCCN(CC)C3)=O)C2)C1 C(C)(C)(C(C)NC(=O)C(c1cscn1)N(C)C)OC c1(N2CCN(Cc3c(OCCCC)cccc3)CC2)cncc2nnnn12 N1(C(C(CC)=CC)=O)CCC(C(F)CNC(=O)CN2CCCCCC2)CC1 C12(C(=O)NC3CN(C(CCCOCCOC)=O)C(C)(C)C3)CCC(N=[N+]=[N-])C1C2 N1(C(CC(CCOC)(C)C)=O)CC2CN(C(=O)CC(C)F)CC2(C)C1 CC1(C)CCC(C(=O)Nc2ccc(Cl)c(C#N)c2)CN1C(c1cccnn1)=O N1(C(=O)NCCC(C(C)C)N2CCCC2)CCc2ncccc2C1 C1(C(N2CC(O)(C(C(=O)N(CC(C)C)CC)F)C2)=O)COCCN1C O=C(C1CS(=O)(=O)c2ccccc21)NCCCNC(c1cnncc1Cl)=O C1(C)(C(=O)NCC2C(NC(C3CCN(CC)C3)=O)COC2)CC2CC2C1 c1(C(=O)NCCCCC2CN(C(CCOCCOC)=O)C2)occc1Br Cc1nc(C(=O)NC2(CN(C(=O)CCCc3ccccc3)C)CC2)cc(O)n1 C1(OC)CC2(C1)CC(C(=O)N(CC(C)O)CCNC(=O)C(C)(C1CC1)SC)C2 Cc1cccc(CSCC(=O)N(CC(C)(C)NC(C2CC(C#N)C2)=O)C)c1 N#Cc1cnc(N2CCCC(CCNC(C3(O)CC4CCC3C4)=O)CC2)c(Cl)c1 c1(CN(C(=O)CCC2CCN(C(c3cc(CC4CC4)on3)=O)C2)C)nccn1C C(=O)(CCS(=O)(=O)N(C)C)N(C1CCC(NC(=O)C(c2ccc(Cl)s2)=O)CC1)C C1(CNC(CCCC#CC)=O)CC2CCC(C1)N2C(C1(C)CC(C)(C)OC1=O)=O C(=O)(CCCC(F)(F)F)NC(C(C)O)C(=O)NC1CC2CCC1C2 C(=O)(C(C(=O)N1CC2CC(NC(=O)C=Cc3nccs3)C1C2)C(C)C)OCC Cc1cnc(N2CCC(C(C)NC(=O)C3=CC(C)(C)C3)CC2)nc1C C1(NS(CC(C)N)(=O)=O)CC2OC(=O)CC12 c1(C(=O)NC2CC(F)CN(C(=O)CC3CCCC3)C2)cccc2c1COC2 c1(C(N2CC(NC(c3ccc(C)nn3)=O)CC2(C)C)=O)cccc2ccncc12 C1(C)(CNC(C(C)N(C(C2CC(CC)C2)=O)C)=O)CCCO1 C1(NC(c2c[nH]c(=O)cn2)=O)CN(C(=O)CCOCC2CCC2)C2(CCCC2)C1 c1(C(N2CC(CNC(C(CC#C)O)=O)(COC)C2)=O)ccc(=O)n(CC)n1 N1(C(C2(C(C)(F)F)CC2)=O)CCCC(F)(CNC(c2ncc(Cl)cc2F)=O)C1 C12(CNC(C=CCC)=O)CCCC1CCN2C(=O)C1=COCCO1 S(=O)(=O)(c1cnc(Cl)nc1)Nc1c(C(=O)NCc2ccn(C)n2)nccc1 c1(C(N(CCSCC(C)C)C)=O)ccc(CC(=O)NC2CC2CF)cc1 N1(C(CCCC)=O)CCN(C(=O)C(C)=C2CCCC2)CC1c1cccc(Cl)c1 C1(CNC(C2CCN(C)CC2)=O)CCCC12CCN(C(c1c[nH]nc1F)=O)CC2 C(C(=O)N1CC(OCCC(=O)NCC2CC2CC(C)(C)C)C1)(C1CC1)SC CC1CCC(NC(=O)C(F)C2CCCC2)CN1Cc1ccccc1Cl CCC(C)(C)C(O)C(=O)N1CC(COC)(NC(c2sc(N(C)C)nc2Cl)=O)C1 C1CCN=C2N=C(C=CN2)N1C.c1(OC)cnc(Cl)cc1COC(C)(C)C c1(C(N2CCCN(C(c3ccc(C(C)C)cn3)=O)CC2)=O)ccc2nccn2c1 N1(C(C(C)OC2CCCCO2)=O)CC(C2CN(C(=O)COC3CCCCC3)C2)C1 c1(C(=O)NC2CN(C(=O)Cc3ccnnc3O)C2)cc2c(nn1)CCC2 C#CCC(O)CC(=O)NC1(C)CCN(C(c2cncc(N3CCCC3)n2)=O)CC1 C(=O)(C1=C(C(C)=O)N(CCF)C(=O)NC1c1cc(C)nn1CCO)OC C=CCCCC(C(=O)NC1CC1)N1CCC(Cc2cnn(C)c2)C1 c1(OC)ncc(C(N2CCC(NC(c3cscc3OC)=O)C(CO)C2)=O)cc1Cl c1(NCC)ncc(C(=O)NCCCCNC(=O)C(C(C)C)NC)cc1Cl N1(C(C2C=CCN(C(CC=CC)=O)C2)=O)CC2(C1)CC(C)(C)C2 Nc1c(F)cc(C(=O)NCC2CCCCCN2C(=O)C(O)C2CC2)cc1F CCCCC(C(=O)N1CC(NC(c2nc(C)oc2OC)=O)C1)N(C)C N1(C(C(CC#C)O)=O)CCC2CN(C(=O)CCC(=O)c3ccccn3)CC12 C1(CNC(C2(C(C)NC(C(CSC)C)=O)CC2)=O)CCCN(C)C1=O C=CCCC(O)CN(C)C(C1(CNC(c2cc(C(F)F)[nH]n2)=O)CC1)=O C1(C(N2CCC(C(C)(C)NC(CC3COCC(C)O3)=O)C2)=O)CCCCC1(C)C C1(N(C(c2cccc(SCC)c2)=O)C)CN(C(c2c[nH]nc2C)=O)CCC1O Nc1cc(C(N2CCN(C(c3coc(CO)c3)=O)CC2C2CC2)=O)cc(F)c1O C1(C(=O)NCC(=O)NCc2cc(C(C)C)on2)C2(CC2)C12CC2.C1(=O)CN1 C1(C(=O)NCC2(OC)CN(C(=O)C(C)O)C2)Cc2cccc(C)c2O1 C#CC1CC2(CC2)CN1C(C1CC(NC(=O)CC2CC2CC)CCO1)=O c1(C(=O)NCCN(CCOC)C(C2CCC(=O)N2)=O)cc2cccn2c(O)n1 S(=O)(=O)(c1ccc(NCCCN2CCCC2=O)c(F)c1)N1CCC(OC)(CO)C1 c1(C(N(CC(CC)NC(c2ccccn2)=O)C)=O)cccc(CC2CC2)c1 N1(C(C2CCC(C)(C)C2)=O)CC(NC(=O)CN2CCOCC2)CC(F)C1 c1(OCC(C)OC(C=CCCC)=O)cc(C)nc(-c2ccccc2)n1 N1(C(C2CC(CC)C2)=O)CCC2C(C(N3CCC(C(N)=O)(N(C)C)C3)=O)C2C1 C1(C(=O)NCC(=O)NC)CCCN(C(=O)C=CC2CC2)C1 N1(C(c2nc(C)sc2C)=O)CCCC12CN(C(=O)CSc1cccc(F)c1)C2 C(=O)(C1CCCc2scnc21)N1CCC(NC(=O)CS(=O)(=O)C2CC2)C12CCC2 c1(C(N2CC(O)(CNC(C(C=C)O)=O)C2)=O)cnc(-c2ccoc2)[nH]c1=N N1(C(CNC(=O)OCC=C)=O)CC(NC(C2(CSC)CCOCC2)=O)C2(CC2)C1 C12(NC(C(c3ccc(OC)cc3)O)=O)CCC(CC1)N(C(C1CC=CCO1)=O)C2 N1(CCN(C)C)CC2(C1)OCc1cc(-c3ccc(F)c(OC4CCC4)c3)ccc12 CC(C)(C)CC(=O)N1CCCCC1C(N1CCOC(CCN(C)C)C1)=O CC1(C)CCCC1CCNC(C1CCC(CNC(=O)C(F)=CC2CC2)C1)=O c1(NC(Cc2nccc(OC)c2C)=O)cc(SC(C)(C)C)cc([N+](=O)[O-])c1 N1(C(=O)OC(C)(C)C)CCCC2CC12CNN1CCCCCC1 CC(C)C(C#N)C(=O)NC(C(=O)N(C1CC2CC2C1)C)C(C)(C)O Cc1c(C(=O)NC2CN(C(=O)CC3CCS(=O)(=O)C3)CC2C)ccc2cncn12 c1(NC(CC(C)C)CNS(C)(=O)=O)nccc(=NCC2CCOC2(C)C)[nH]1 c1(C(=O)N)cccc2ccncc12.CC(C)(C)CC(F)C(=O)NCCCC=O C(=O)(C1CCOc2ccc(F)cc21)NC1(CNC(C2CCCO2)=O)CCOCC1 C1(NC(c2c(C)ncs2)=O)CC2CC(C1)N(C(c1ccnc3c1CCO3)=O)C2 C(=O)(CCCC(F)F)N1CC2C(CNC(CCC(C)N(C)C)=O)(C2)C1 C(CCCC(=O)NC(C1CCOC1)CO)NC(COCCCC(C)C)=O CC1C(NC(COC2CCCC2)=O)CCCN1C(=O)COC1CC2CCC(C1)C2 C=C(C)CCCC(=O)NC1(C(=O)NC(c2ncccc2F)C)CCC(C)(C)C1 c1(CC)c(-c2nc(CCO)nn2CC(F)(F)F)cnn1C(C)CC C1(CC(N2CCC(CN(C(c3cnc(C)nc3)=O)C)C2)=O)CCCCC1(F)F c1(C(N(CCC)CCNC(C2CCC(=O)N(C)C2)=O)=O)c(F)cc(C#N)cc1F c1(CNC(Cn2cc(C(C)O)nn2)=O)ccc(OCc2ncccc2C)cc1 C1(NC(c2c(CC)occ2)=O)CCC(N(C)C(C2CC2CCOC)=O)CC1 c1(C(N2CC(NC(C3C(OC)CCCC3)=O)C2)=O)ccc(C)c2c1NCCC2 C(C(C(=O)NC1(n2ccnn2)CC1)NC(C1(C(=O)C2CC2)CC1)=O)OCC c1(C(=O)OC)cnn2c1CC(NS(=O)(=O)CC(C)(C)CCl)CC2 n1(C(CC)C)ncc(C(=O)N(CC(C)N(C)C(C2CC2CC(C)(C)C)=O)C)c1C N1(C(c2cc(CSCC)on2)=O)CC2CN(C(=O)C(c3scnc3C)O)CC2C1 c1(OC)c(C(=O)N(CC2CC2C)CC2CC2)cccc1F N1(C(CC=CC)=O)CCC2CN(C(c3c(CC)nn(C)c3CC)=O)CCC2C1 N1(C(C2(C(=O)OCC)CC=CC2)=O)CCC2(CCC2)C(CO)C1 c1(C(N2C(C)(C(N3CCCC(OCC)C3)=O)CC2)=O)c(F)ccc(C)c1F c1(CNC(C(N2C(COC)COCC2)c2cn(C)nc2C)=O)ccc(C)cc1Cl c1(C(=O)NC(CCOC)CNC(=O)C(C)(C2CC2)OC)c(N)cc(F)cc1Cl C1(C#N)(CNC(CC2(C)N(C(c3cc(OC)n[nH]3)=O)CC2)=O)CCOCC1 C=CC(CC)CC(=O)NC1CCC(CC(=O)N(C)CC2CC(=C)C2)C1 Cc1[nH]c(=NCc2ccc(C(F)(F)F)nc2)sc1C(=O)Nc1c(O)n[nH]c1C N1(C(C(C)n2ccnc2)=O)CC(NC(=O)C=Cc2c[nH]cn2)C(C)(C)C1 N1(C(c2ccccc2Br)C(=O)NC2(C)CC2)CCCC2(CCC2O)C1 C(CCC(=O)N(C1(C(N)=O)CCC1)C)N(C(C)C)C(=O)SC1COCCO1 c1(CC(C(=O)NCCC(C)(C)NC(=O)CCCOCC#N)O)c(F)cccc1Cl c1(OC)nc(Cl)c(C(=O)NC2CN(C(=O)Cc3csc(C(C)C)n3)CC2SC)s1 c1(CC(=O)N(CCCCN(C(CSCC(=O)OC)=O)C)C)ccn(C(C)C)n1 c1(CC(=O)NCCN(C(C)=O)C)coc2ccc(C)cc12 C(=O)(NNc1ncc(C#N)c(OC)n1)N1CCC(OCC)(OC)CC1 S(=O)(=O)(c1ccc(=NCC2(F)CC2)[nH]c1)NCC1CCCC(SC(C)(C)C)CC1 CC1(C)CC1(Br)C(=O)NC1CCC(NC(c2cn(CCO)nn2)=O)C1 C1(CCNC(C=CSC)=O)CN(C(=O)C(C)NC(c2cccs2)=O)CCO1 C(=O)(C(O)(C(F)(F)F)C1CC1)NCC(CNC(c1n[nH]c2c1CCC2)=O)CO C(CCN(C(=O)C(C)=CC1CC1)C)(C(C)C)NC(C1(C=C)CC1)=O c1(NCc2cnc(Cl)s2)cccc(OC(F)(F)F)c1F.C12CCC(CC1)C(=O)N2 C(=O)(C(C)(C(C)C)OC)NCCC1N(C(c2ccc(OC)s2)=O)CCC1 C12(NC(COCCC)=O)CCCC1CN(C(C13CC(CN1C1CC1)C3)=O)C2 N1(C(C2CN(C)C(=O)N2)=O)CC(N=c2cc(C(C)(C)C)nc(Cl)[nH]2)C2(CCC2)C1 Cc1nn(C)c2ncc(C(N3CCC(C)C3CNC(=O)C(C)CF)=O)cc12 C12(C)CC(C1)NC(=O)CCN(CC)CC=CC(=O)NC2.C(C)(=O)OC CCCCC(C)CCC(=O)NC1CC(C)(NC(c2cncc(C=C)c2)=O)C1 C1(C(N2C(CC)CC(C)C2)=O)N(C(=O)C=Cc2ccnn2C)CCC1(C)C c1(C(=O)NC2CCCN(C(C(CCC)C)=O)C2)ccc2ccccc2c1C Cc1nc(C(=O)N(CCC#N)CCN(C)C)sc1-c1ccc(C(F)(F)F)nn1 CC1C(NC(c2cnc(Cl)[nH]2)=O)CCCN1C(c1ccc(-n2cnnn2)cn1)=O c1(NC(C(CNC(C(CC)(F)F)=O)CC2CC2)=O)cc(C)c(F)cc1O C1(CNC(=O)CCc2ccsc2)CC(F)(CNC(=O)C=Cc2cc[nH]n2)C1 c1(C(=O)NC(C2CN(C(C3CCCC(C)CC3)=O)C2)C)cc2n(n1)CCCC2 N1(C(C(C)NC(=O)C2CC2)=O)CCOC(CCNC(c2cccc(N)n2)=O)C1 C1(N(C)C(C2CC2CF)=O)CCC(NC(=O)C=Cc2ccc[nH]2)CC1 c1(CCCC(=O)NC2CCC(NC(c3c(C)nc[nH]3)=O)C2)ccc(F)c(F)c1 C(C(F)(F)C(=O)NC(C1CCOC1)CNC(=O)C(C1CCOCC1)=O)NC(C)=O O=C1CCC2(CCC(NC3CC4(CCCO4)C3)CC2)N1 c1(C(=O)NC23CC(NC(C(C)(O)Cn4cc(Br)cn4)=O)(C2)C3)cccc(Cl)c1F C1(C(=O)NCc2c(C(=O)NCCC3CCN(C)CC3)n[nH]c2)CCCC12CCC2 c1(N(CCCC)C)ccc(S(=O)(=O)NCc2ccc(OC)c(OCC)c2)cc1Br c1(NC2CN(C(C(=O)Nc3c(OC)cccc3)=O)CC2C)ccc(Cl)c(Br)c1F c1(C(C)C)cc(F)c(NC(c2ccc(N3CCCCC3=O)cc2)=O)cc1F N1(C(c2cc(CC)[nH]n2)=O)CCC(C(C)(C)C)(CNC(=O)COC2CCOC2)C1 C1(C)(C(N2CCCN(C(C)=O)C2)=O)CC(O)CN1C(c1ccn(C)n1)=O c1(C(N(CC(C)CNC(C2(C(F)F)CC3(CC3)C2)=O)C)=O)nn(C)c(Cl)c1Cl C1(=CCNC(=O)CC2COCC2O)CCN(C(C2COC(=O)O2)=O)CC1 N1(CC(N2C(c3cn(-c4ccc(C)cc4C)nn3)CCC2)=O)C(=O)OC(C)(C)C1=O c1(C(=O)OC)cc(C(=O)NCC2CN(C(C3CC(C)=NO3)=O)CCO2)n(C)c1 C(C(C)(C)CNC(=O)Cc1cscn1)N(C(=O)C(F)(F)c1ncccn1)CC N1(C(C2(F)CCN(C(c3cc(OC)n(C)n3)=O)C2)=O)CCCC(O)C1C C(=O)(CCCC(C)(C)C)N1CCC(C(=O)NCCN(CCO)CC)(CC)C1 C(=O)(CCC(C)CCCC)NC(CNC(c1ccc(C=C)cc1)=O)(C)CC CN1CCCC1(C)CC(C(=O)NCC(F)F)N1CCC(C(=O)NCC2CC2)C1 n1(CCC=C)c(N(CCc2ccc(Cl)cc2)CC)nnc1CC1CCCCC1 C1(C(N2CC(C(C(=O)NCCC3CC(OC4CC4)C3)O)C2)=O)CC12CCCC2 N1(C(C(=O)N(C)C)=O)CCC(C=CC(=O)N(C(C2CCOC2)CO)C2CC2)CC1 c1(C(C)=O)ccc(CC(=O)NCCCCCNCC2CCC(c3ccccc3)C2)s1 CCCCC(CC)CC(=O)N1CCCC(O)(CN(C)C(c2ccn(CC)n2)=O)C1 c1(OC)ccc(CC(N2CCN(CCCNC(=O)CS(N)(=O)=O)CC2)=O)c(F)c1 C(=O)(C(C(C)CC)NC(=O)CC1CC1(C)C)NCc1nc(CC)oc1 N1(C(C2C(=C)C2)=O)CCCC1CN(C(=O)CCc1ccccn1)CC(O)CC c1(N2CC(C)C(c3c(C)c(C)[nH]n3)C(C)C2)nc(Cl)nc2c1ncn2C CC1(C)C(NC(=O)CCOc2cccc(C#N)c2)CCN1C(=O)COCC1CC1 C(=O)(C1=C(Cl)CCC1)N1C(C)(C(=O)NCC(CCCC)O)C=CC1 C1(C(N2C3(CN(C(=O)Nc4cc(CC)on4)C3)CC2)=O)CCCN2CCCC12 c1(CCC(=O)OC(c2csc(Br)c2)C)nnc(C2CCCC2)o1 C1(NC(c2c(C)nccn2)=O)CC(O)CN(C(C2C3CCCCC23)=O)C1 C12(CNC(c3cc(OC)c(Cl)cc3)=O)CCCC1CN(C(C1CCSC1)=O)C2 C1(n2cnnn2)(C(C2CCCO2)NC(=O)Cc2nc(C(=O)O)cs2)CCSCC1 C1(CNC(c2cc(C)ncc2C)=O)CN(C(=O)CC2CCCO2)CC(C)(C)C1 C=CCC(CNC(c1ccn(C)n1)=O)NC(c1cn(CC2(C)COC2)nn1)=O CC1CN(C)CCCN1C(C1C(C)CN1C(=O)C1=CCCCCC1)=O C(C(C)(C)CC(=O)N=c1ccn(C)[nH]1)NC(C1(C)CN(C)C(=O)C1)=O c1(C(N(CC(O)CN(C(=O)C(C)(C)C)C)C)=O)[nH]cnc1C#N.N12CCC1C2=O Cc1ccc2nc(CNC(=NCCCC#C)NCC3CCOC3)cn2c1 c1(C(C(=O)NCC2CC2)N(C(c2cc[nH]n2)C(=O)OC)CC)ccccc1Br C=CCC(CC)NC(c1snnc1C)c1nnnn1CCN1CCOCC1 C1(C(N2C(CNC(c3c(C)cc(C)s3)=O)CCCC2)=O)CC(S(C)(=O)=O)C1 c1(CNC2CC(CC(N3CC(O)C3)=O)C2)c(O)ccc(F)c1F c1(CNC(C(N2CCC(NC(CCC)=O)C2)=O)=O)cc(Cl)c2c(c1)OCO2 CCC(C)C(O)CC(=O)NCC1CCCCC1C(N1CC(CC(N)=O)C1)=O n1(C(C(=O)OC)C)nnnc1C(c1cnn[nH]1)NC(C)COCCOC C1(C)(C)C2CC(C(OC)C(=O)N2)CN1C.C(=O)CC(C)OC.CO O=C(CCC(=O)N1CCOCC1)NC1CCN(C(c2coc(Cl)c2)=O)CC1 C1(C(=O)NC(CCCNC(c2c(C)n(C)nc2)=O)C)CCCNS1(=O)=O S(=O)(=O)(c1ccc(C(N2CC(CNC(=O)CSC)CC(C)(C)C2)=O)cc1)NCC Cc1cn(C)cc1C(N1CCC(CO)(CNC(C2C3COCC23)=O)C1)=O C(CC(=O)N1CCC(N(C)C)C(C)(C)C1)(C(F)(F)F)OC.C1(=O)C(C(C)C)N1 N1(C(CC(COC)(C)C)=O)CCC2(CCCN(C(C3CC3C)=O)C2)CC1 CC1CC(=O)NC(C(N2CCC(C)C2C(=O)NC2CCC(N(C)C)C2)=O)C1 c1(C(=O)NC2CCCN(C(CC(=C)C)=O)C2)c(F)cc(F)cc1F N1(C(CC=C=C)=O)CC2CC(NC(C3CCN(Cc4ccccc4)C3)=O)CC1C2 C12(NC(c3c(OC)cccn3)=O)CCOC(CNC(=O)C(C)n3cccn3)(C1)C2 C1(NC(Cc2cc(C(C)C)no2)=O)CCN(C(C2CCS(=O)(=O)CC2)=O)CC1O C(=O)(C(C)CC(=O)NC(CC)CN(C(=O)C1=COCC1)C)OC c1(CCC(=O)NCC23C(CN(C(C4ON=C(CC)C4)=O)C2)C3)ccc(C)c(C)c1 N1(C(C(C)(C)c2cccs2)=O)CCCC2(CC(NC(=O)Cc3cnns3)CO2)C1 c1(OC)ccc(C(=O)NCC2CCN2C(C2(OC)CCSC2)=O)cc1S(C)(=O)=O c12cc3c(cc1F)CN(N1CC4(CN(C)C4)C1CCC2)CC3.CO N1(C(CC2CC(OCC)C2)=O)CCCC1C1CC1.C1C(C)(C2CCC2)NC1 C1(C(=O)NCc2cn(C3CCN(C(C=C)=O)CC3)nn2)CCC2CCCCN12 c1(C(=O)NC2(C(=O)NC(C(C)F)C)CCCC2)cnn(C)c1C#N c1(C(N2CC(NC(C3C(CN(C)C)C3)=O)C2)=O)ccnc(N2CCC2)c1 N1(C(C(C)C)=O)CCC(C(C)(C)C(=O)N2CCSCC2)C1 CCCC(C)(O)CC(=O)N1CC(OC)C(NC(c2csnc2C2CC2)=O)C1 C1(NC(C2(COC)COC2)=O)CC2CC(NC(=O)CC3CCOC3)C1C2 c1(C(=O)NC(CCCNC(CCNC(=O)OC)=O)C)ccc(CCF)cc1 N1(C(C2CCC(N(C)C)C2)=O)CC2CC1C2CNC(c1ccc(C(N)=O)o1)=O C#CCCC(C(=O)N(C)CC)NC(=O)C(C)N(C(CC)CC)CC Cc1cc(CC(=O)NC2(C3CCCN3C(C3CC4CCC3C4)=O)CC2)cc(C)c1 C1(c2nccc(CN(CCOC)C)n2)CCCCN1C(C1C2CCC(=O)C12)=O C1(C(=O)NC2CN(C(C(CC=C)CC)=O)CC2C)CCC2(CCCC2)CC1 C(N=c1nc2scnc2c(N2CCC3(CC2)CCN3C(N)=O)[nH]1)C1(N(C)C)CC1 N#CC(F)(F)CCC(=O)N(c1ccncc1)CCN1CCC(N)CC1 c1(C(=O)NC(C2CCCN(C(=O)C(=C3CCCCC3)F)C2)C)cc(N)cc(O)c1 c1(CNC(=O)NCC(C)CN2CCOCC2)cccc(CC2CCC2(F)F)c1 C1(NC(c2cc(CC)oc2C)=O)CC(C(=O)Nc2csc(C)c2)C12CCC2 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC1C(C)CN(C(=O)CCC#N)C1 CCC(CC(=O)N1CC(OC)CC1CO)NC(=O)COCC(=O)OC C=CC(C)(C)CC(=O)NC1(COC)CCN(C(c2cc(F)cs2)=O)C1 c1(OCC)ccc2cc(C(N3CCC(NC(C4C(C)C4C)=O)C3C)=O)[nH]c2c1 CC1CN(C(c2cncc(C(F)F)c2)=O)CC1CNC(c1cnc(C(C)O)s1)=O C1(CCC)CCCN(CCC2(c3ccccc3)CCCC2)C1.C1CN1 c1(C(N(C2C(C)CC2)C)=O)ccc(NC(N)=O)cc1 C1(NC(CCC)=O)CCC2CCN(C(c3ccoc3Cl)=O)C12 c1(C(N2C(CNC(c3cnco3)=O)CC2)=O)cnn(CC2CC2)c1 O=S(=O)(c1ccc(N2CCOC(CCF)C2)c(F)c1)NC1COC2(CCCC2)C1 c1(C(=O)NC2C=CC(CNC(C3(CC#C)CCOC3)=O)C2)cc(Cl)c(N)cc1F CC(C)CC(F)C(=O)NCC(C(C)(C)C)NC(c1cn(CC(F)(F)F)nn1)=O CC1(C)CCC(O)(C(=O)NCC2CC2NC(C2(c3cccs3)CC2)=O)CC1 N1(CC2(N3C(=O)NCCC3)CCC2)CCN(C(=O)C=CCBr)C(=O)C1 CCC(C)C(O)C(=O)NCC(C)CNC(C1(O)CCCCCC1)=O c1(C(=O)NCC2(CNC(C(CCC)C)=O)CCCCC2)cncc2c[nH]nc12 C1(=CC(=O)NCC(c2c(F)cccc2F)NC(CC)=O)CCCCC1(C)C c1(SC)nc(CC(=O)NC(c2ccc(C)cc2)C2CCC2)c2ccccn12 c1(OC)nc(C(=O)NC2(CNC(=O)CC3CC(SC)C3)CCCCC2)sc1C C(C)(CNC(c1cn(C(C)C)nn1)=O)(CC)NC(C1(SC)CC1)=O C1(CNC(CC(CC)C)=O)CN(C(=O)COCCCF)CCN1C c1(C(N2C(CCNC(CS(CC)=O)=O)CCC2)=O)cnc(O)c2cncn12 N1(C(C(C)OCCCC)=O)CC2CC2(NC(=O)CNS(=O)(=O)CC)C1 S(=O)(=O)(c1cc(Br)ccc1Cl)N(C(c1cnn2ccccc12)=O)CC1CNC1 c1(CC)cccc(F)c1C(N1CCN(C(=O)CCC(C)(F)F)CC1CO)=O C1(NC(C2ON=C(CC)C2)=O)CN(C(c2c(Br)n[nH]c2C)=O)CCC1O c1(C(c2nnnn2-c2ccccc2)NCCCCCS)ccncc1.CC(C)(C)O N1(C(Cn2c(C)ccn2)=O)CCCCCC(NC(=O)CCN2CCCC2=O)C1 C1(CNC(c2c(C)ncs2)=O)CN(C(=O)CC2(C(F)(F)F)CC2)C2CC12 C(=O)(CCC(=O)c1cccnc1)N1C(C(N(CC(N)=O)C)=O)CCC1 C(=O)(C#CC1CC(F)(F)C1)NCC=CCNC(c1c(C)ncc(Br)c1)=O N1(C(C2(CNC(C(C(C)C)F)=O)CCCO2)=O)CC23CCC2(COC3)C1 C(=O)(C(CCF)N(C(=O)COC)C)N(CCCn1ccnc1)C.c1(OC)ccccc1 CON(C)CCCNC(=O)C(c1ccoc1)NC(C1CC=CCC1)=O c1(SCC)ccc(C(=O)NCCCC(C)(C)NC(c2cncc(NC)c2)=O)cc1 N1(C(c2c[nH]c(=N)o2)=O)CC(CNC(=O)C=Cc2cccs2)OC2(CCC2)C1 c1(OC(C)=O)ccc(Cl)c(CN2C3CCCC(C3)C2CN2CCC(Br)CC2)c1F N1(C(c2c(C)ccs2)=O)CCCC(CN(C(=O)C(C)OC2CCOC2)C)C1 C1(C(N2C(COC)CN(C(c3cc(C)no3)=O)CC2)=O)CCC2(CCOCC2)C1 C(C(=O)NCC(c1ccc(C)cc1)NC(C1(C)CC=CC1)=O)(C(C)C)OC c1(CNC(c2c(C)cco2)=O)ccc(CNC(C2CCOC(C)C2)=O)c(F)c1 c1(OC)cc(OC)cc(NC(C2CC3(CC3)CN2C(c2ccc(O)nc2)=O)=O)c1 N1(C(CSSC)=O)C2CCC1CC(NC(c1cnn(C)n1)=O)C2 N1(C(C2C(C)=CCS2)=O)CC2CCC(Nc3ncnc(Cl)c3CO)C2C1 C12(NC(C(C3CCOC3)OCC)=O)CC(C1)N(C(=O)C=Cc1csc(C)n1)C2 CC1CN(C(=O)C(CCF)NC(C2CCC(O)CN2C)=O)CC(C)(C)O1 c1(C(=O)NCC(C)(C)NC(C2CC(C)=C(C)CC2)=O)cc(C)c(C)c(F)c1 C(=O)(C(Cn1cccn1)C(=O)N1CCC(O)(C(c2ccccc2)O)CC1)OCC Cc1cc(F)c(S(=O)(=O)N2CCC(c3nc(C)c(C)s3)C2)c(Br)c1 Cc1cc(N)n2ncc(C(=O)N(C)CCNC(=O)CCC3CCCN(C)C3)c2n1 CC(C#N)CN=c1nc(N2CCOC(CCF)C2)c2c([nH]1)CCOC2 CC(C)CC(CNC1CC(n2ccnc2)C1)N(C)C N1(C(c2n(C)nc(Br)c2)=O)CCC(c2ccc(F)cc2)C(N)C1 N1(C(c2ccc(C)c(CO)c2)=O)CCC(C2CC2)(CNC(=O)C(C)NC(N)=O)C1 c1(C(=O)NCC2CC(COC)CN2C(=O)CC2CCOCC2)cccc(C)c1O C1(NC(=O)C(=Cc2c[nH]cn2)F)COCCN(C(=O)CC2CC(O)C23CCC3)C1 N(C1CCc2ccc(Br)cc21)C(C1(C)CCN1C(c1cc(F)cc(Br)c1F)=O)=O C1(CC)CN(C(=O)CSc2ccc(C)cc2C)CCN1C(c1cnn[nH]1)=O c1(C(=O)NC(CNC(C2(CCC)CCC2)=O)C2CC2)ccc(CC)nc1 c1(CSCC(=O)NCC2(O)CCN(C(=O)CC(F)F)C2)ccc(F)cc1 Cc1cc(N2CCOCC2)nc(N2CCCC2CNc2ccc(Br)o2)n1 C(=O)(C(O)P(C)(C)=O)NC(CCOC)C(=O)NCc1cc(F)cc(F)c1 C1(COC(c2onc(C)c2C)=O)CN(C(=O)OC(C)(C)C)C2CCN1C2 CCC(O)C(C)C(=O)N(CCCCCC(=O)NC1COCC1F)C O=C(C1=NNC(C(F)(F)F)C1)NCC1CN(C(c2ncccn2)=O)CCO1 C1(NC(c2cn(CC)nc2)=O)CC2CC1N(C(c1nnn(C)c1N)=O)C2 C1(N(C(=O)CC2CC(N)C2)C)CCN(C(N)=O)CC1.c1(C=O)c[nH]c(C(N)=O)c1 C(c1ccc(F)cc1F)=CC(N1CCN(C(CSc2ccc(C)cc2)=O)C2C1C2)=O N1(C(C(C)O)=O)CCCC(O)(CN(C(=O)C(O)c2ccco2)C)C1 c1(C(N(C(C)CNC(C2(N3CCOCC3)CC2)=O)C)=O)cnn2cccc(Cl)c12 c1(OC(C(N2CC(CNC(c3cc(C)sn3)=O)OCC2)=O)C)ccc(F)c(F)c1 C1(NC(c2cn(CCOC)nc2)=O)CC2C(NC(=O)CN(C)C(=O)C3CC3)C2C1 Cc1oc(C#N)cc1C(N1CCCCC1CC(=O)NC(c1cncs1)C)=O C1(C(=O)NC2CCC3(CC3)C2)CC1C1CN(C(=O)C=Cc2ccoc2)C1 n1(SCC)nc(C)c(CC(C)C(=O)NC2CC(NC(C3(C#N)CCC3)=O)C2)c1C CCC1=C(C(=O)NCC2(F)CN(C(c3ncnc(C)c3C)=O)C2)SCCO1 C1(C(=O)NC(C(C)C)CCN(C)C(c2ccc(CF)cc2)=O)CCC(C#N)CC1 CC1(C(=O)NCC2CC2C2CC2N)CCC(=O)NC1 C1(CC=C)(NC(=O)Cc2cc(F)cc(Cl)c2)CCN(C(C2CCCCO2)=O)CC1 C(=O)(C(C(C)C)NC(C)=O)NCCCC(C)NC(c1c(SC)ccs1)=O C12(C(=O)N(CC3C(NC(c4c(C)noc4C)=O)C3)CCO)CCC(C1)OC2C C(c1ccc(OC)cc1C)=CC(N1CC(NC(C(C)OC)=O)C(C(F)(F)F)C1)=O c1(N(C(c2ccc(OCC#C)cc2)=O)CC)nc2cc(Cl)ccc2o1 N1(C(c2c(CC)nn[nH]2)=O)CC(C(=O)NC(c2ccoc2)C)C(C)(C)C1 C#CC(C)(C)C(=O)NCCCOCCCNC(=O)CC1CCCN1C c1(C(=O)NC2C=CCN(C(Cn3c(C)nnn3)=O)C2)ccc2ccccc2c1F c1(C(N2CCC(O)(CN(C(c3nc(C)n(C)n3)=O)C)C2)=O)ccc(Cl)nc1O CC(C)CC(C(=O)NC1CCCN1C(=O)CCNC(N)=O)NC(=O)OC(C)(C)C c1(C(C(=O)NC(CC)(C)C)N(C)C(c2ccc(F)cc2)C)sc([N+](=O)[O-])cc1Cl c1(C(N2CCC(CC=C)(NC(=O)C(C3CC3)OCC)C2)=O)cc(N)cc(F)c1 N1(C(CCCCCSC)=O)CCC2CCCN(C(=O)Cc3c[nH]nc3C)C2C1 c1(C(=O)NCC2=CCN(C(c3cc(C)ns3)=O)CC2)nc[nH]c2nccc1-2 C(C)(CCC(=O)N1CCCCC1CNC(C12CC(C(C)C)(CO1)C2)=O)OC N1(C(C(CNC)C)=O)CCC(C(=O)NC2(C3(OC)CCC3)CC2)CC1(C)C N1(C(c2cccc(NCc3c(OC)cc(C)cc3)c2)=O)CCC2CC(=O)NC2C1 C1(N(C(=O)Cc2n[nH]c(=N)s2)CCC)CCN(C(=O)CCNC(=O)CC)CC1 c1(C(=O)NCCCCCN(C(=O)CC2(O)COC(C)(C)C2)C)cccc(=O)n1C c1(NC(c2c(C)noc2)c2nnnn2C2CCCCC2)cncc([N+](=O)[O-])c1 NS(=O)(=O)c1cnn(CC(=O)NC2CCCCC2NC(=O)C(F)(F)CO)c1 C1(NC(C(CCCC)O)=O)C2CCCC1CC(C(N(CC(=O)NC1CC1)C)=O)C2 CC1OCCC1CC(=O)NCCN(C(=O)COCP(C)(C)=O)Cc1ccccn1 c1(C(N(CC(CNC(C(N2C(CC)CCC2)=O)=O)O)C)=O)ccc(C(C)C)cn1 C(CC(=O)NCc1cccc(C#N)c1)(C(C)(C)C)NC(C(C)n1ccnn1)=O C1(C(=O)NCC(C)O)CC(F)CN1C(=O)C(c1cccc(Br)c1)O C1(CC(=O)NCC2CC(=C)C2)C2CCCC2N1C(=O)CC1CNC(=O)C1 C1(NC(c2cccs2)=O)CC2CCC(C1)N2C(=O)CCc1cc(F)ccc1F N1(C(C(C)OCCC=C)=O)C2CCC1C(C(=O)NCC1CCCOC1)C2 C1(CC(=O)NC(CNC(CN(CC)CC)=O)CO)CC=CCC1 N1(C(CC(=O)NC2CC2)=O)CCN(C(c2csc(C#N)c2)=O)CC1CCSC1CC1 c1(Cn2cc(-c3scc(C(=O)O)n3)nn2)cccc(Cl)c1Cl C(=O)(C1=CCc2ccccc21)N1CCC(N(C(=O)Cc2cn[nH]c2)C)C2(C1)CC2 CS(=O)(=O)c1ccc(C(N2CCC(CO)(NC(C3CCCOCC3)=O)CC2)=O)[nH]1 N1(C(CC2C(CC)C2(F)F)=O)CCCN(C(=O)Cc2cncnc2)CCC1 Cc1c(C)c(=NC(=O)C(=O)c2cc(-c3cc(O)ccc3F)ccn2)[nH]n1C n12c(nc3ccccc13)C2.CC1CC(C(=O)N(C)C)CN(OC(F)F)C1 C1(NC(c2ccc(C)cn2)=O)CC(NC(=O)CCCSC(C)(C)C)C12CCC2 C(=O)(C(CC)C(=O)N1CCC(C)CC1C(=O)NCC1(C)CC1)OCC CN1CCC(C)(C(N2CCC2CNC(=O)Cn2ncc([N+](=O)[O-])n2)=O)CC1 O=C(C1CC(O)c2ccccc21)NC1CCC(CNC(=O)C(F)C2CCCC2)C1 c1(C(=O)NC(C)CCCCNC(=O)CC2CCOC2=O)cc2ccc(F)cc2s1 CN1CCC(Cc2cn(C3CCCN(C(c4ccncc4Br)=O)C3)nn2)CC1 C1(C(=O)NCC(CC)NC(c2ccccc2[N+](=O)[O-])=O)CC2(CCOCC2)CO1 C#Cc1ccc(CC(N2CCC(C)(NC(C3CC(=C4CCC4)C3)=O)C2)=O)cc1 C1(NC(c2ncn(C(C)C)n2)=O)CC(C)N(C(=O)Cc2cnsc2)C1 c1(C(N(CCCN(C(=O)CN2CC(=O)N(C)C2=O)C)C)=O)cccc2c1COC2 c1(C(N2CCC(CNC(C(C)=CC)=O)CC2)=O)ccc(N)cc1[N+](=O)[O-] c1(C(N2CC(N(CCO)C(=O)C3CC3)C3(CC3)C2)=O)cnc2ccccn12 CON(C)C(=O)Cn1cc(-c2cccc(C(F)F)c2)nn1 N1(C(c2cscc2C2CC2)=O)CCOC(COc2ccccc2)C1 C(=O)(CCCCC(F)F)N1CC(N(C(=O)CC2CC3(CCC3)C2)C)C(C)(C)C1 N1(C(C=CC(C)NC(C2CCCCN2C)=O)=O)CC2(CCOCC2)C1 C(c1ccccc1)=CC(=O)NC(C(c1ccccc1)NC(C=C(C)Cl)=O)C(C)C C=CC(C)(C)CCN=C(NC(C1CC1)C1CC1)N1CCC(O)C(CO)C1 C1(CNC(C(c2n(C)ncc2)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CC1(Cl)Cl c1(C(=O)OC)ccc(C(N2CCCC2Cc2ccccc2F)=O)n1C C#CCC(O)C(=O)N1CC=CC1C(C1CC1)NC(=O)Cc1cccc(C2CC2)c1 CC(=O)CCCC(=O)NC(C(=O)N(C(C)CC(F)(F)F)C)C1CCCC1 c1(OCC)cc(-c2cnc(Cl)c(C(=O)NCCCCO)c2)cc(F)c1F C(c1cncc(F)c1)=CC(=O)NCCC(C)N(C(=O)CCC(=O)N(C)C)C C12(NC(=O)CCn3cnccc3=O)CCC(CN(C(c3cnc(O)s3)=O)C1)C2 c1(C(=O)NCC(C2CCC2)NC(CC(=O)NCC)=O)cc2c(s1)CCC(C)C2 CC1OC(C)CC1C(N1CC2CC1(CNC(=O)C1CC1)C2)=O N1(C(C2(C)N(C(CC(C)C3CC3)=O)CCC2)=O)CC2CCOC2C1 Cc1ncc(C(N2CCOCC(CNC(c3csnc3Cl)=O)C2)=O)cc1N CCCC(C)(C)CC(=O)NC1CC(CCNC(C2(C)CCNC(=O)C2)=O)C1 c12cn(nn1)CC1CC1NC(=O)C21CCC1.c1(C(N(CC)CC)=O)csc(C)c1 C(c1ccc(F)cc1)=CC(C(=O)NC(CCCNC(C=CC=CC)=O)(C)C)=O C=C(Cl)C(C)(C)C(=O)OCN1CCN(C(=O)C(C)(C)N2CCOCC(=O)NC2)CC1 c1(C(=O)NCC2C(NC(c3n(CCC)ncc3)=O)C2)cc(F)cc(Br)c1 c1(OC(c2c(OC)cccc2)=O)ccc([N+](=O)[O-])cc1CN(C)Cc1ccccc1 CC(O)C(C(=O)NC1CC1CNC(c1cc(C(C)(C)C)no1)=O)N(C)C C1(NC(c2c(C)noc2C(F)(F)F)=O)COCCN(C(C23CC2CNC3=O)=O)C1 c1(C(N2CC(CNC(c3c(C)snc3)=O)C3C2C3)=O)cc(N)nc(Cl)c1 N1(S(C)(=O)=O)CC2(C1)C(C(=O)OCc1ccsn1)CCS2(=O)=O C12(NC(c3c(CC)occ3)=O)CCCC1CN(C(C1(CF)CCC1)=O)C2 N1(CCC)CCCCC1C(=O)NC(C)C(CO)NC(=O)C(C)(C)N(C)C N1(C(C2(F)CN(C(CC(C)n3cccn3)=O)C2)=O)CCC2(CCC(O)C2)C1 c1(C(=O)NCC(C)(CO)NC(=O)C(F)n2ccnc2)cn2cccnc2n1 C1(NC(CC(C)C2CCCC2)=O)CC2(CCN(c3ccccc3[N+](=O)[O-])CC2)C1 c1(OC)cnc(C(N2CCC2Cn2cc(-c3c(C)cccc3Cl)nn2)=O)c(Cl)c1 C1(C(N(CC#N)Cc2ccccc2)=O)CCc2ccccc2C1 C1(CNC(=O)CCCC2CCCO2)CCCN(C(C2CC3CCC2CC3)=O)CC1 C1(CCCCC)CCC(C(=O)NC2CCC(N(C(=O)C3=COCC3)CC)CC2)CC1 N1(C(COC(C)C)=O)Cc2ccccc2C(NC(=O)C(C)CS(C)(=O)=O)C1 C1(NC(c2c(C)oc(C#N)c2)=O)CC12CCC(NC(=O)CCN(C)C)CC2 N1(C(Cn2c(C)nnn2)=O)CCCC(C)(C)C1CNC(=O)C=CCF C1(C2CC2)(C(N2CCC(C=C)C2)=O)CN(C(C2CCC(=O)NC2)=O)C1 c1(N2C(C)(CNC(C3CN(C(C)C)C(=O)C3)=O)CCC2)cncc(C#N)n1 c1(NCC2OCC(C)C2)ncccc1S(=O)(=O)NCC1(F)CC(CO)C1 C(=O)(C1OCCc2ccccc21)NC1C(C)CN(C(=O)CCCCCC#N)CC1 c1(C(N2C(CC=C)CCCC2)=O)cc(Cl)c2ccccc2n1 c1(C(=O)NC(CN(C(C(CCSC)NC=O)=O)C)C)cccn2nccc12 N1(C(COC)=O)C2CCC1C(C(=O)NCCC(O)C1CCC1)C2 C(=O)(C1CCCc2c(OC)cccc21)NCCCCC(=O)OCC C1(c2n(CCCOC)nnn2)(NCCCS(C)=O)CCC2(CCC(CBr)O2)CC1 C1(CNC(C(C)(C)CF)=O)CC12CCN(C(c1cnc3[nH]ccc3n1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NCC(C)(C)OCCNC(C(CC)(C)COC)=O C1(NC(C2CC(C(C)(C)C)C2)=O)CCN(C(c2nnc(O)nc2O)=O)C12CCC2 c1(C(=O)NC(C(C)NC(c2ccc(CN(C)C3CC3)o2)=O)(C)C)cc(O)n(C)n1 N1(C(C2C3(CCN(C(c4scnc4C4CC4)=O)C3)C2)=O)Cc2ccccc2C1 C1(OC)C(OC)CN(C(c2cnc(C)o2)=O)C1CNC(C1CCOC1C(C)C)=O Cc1cc(NC(=O)NCC2CC2NC(=O)OCC)nc(S(C)(=O)=O)n1.C(C)(C)(C)O C1(NC(N(CCC)CC2CCCN2Cc2ccccc2)=O)C=CC(C)(C)CC1 CC(C)C(C)(CNC(=O)CNC(c1ccc(Cl)cn1)=O)NC(=O)C=CCF C(=O)(C1CCCc2ccccc21)N1C2CN(C(c3c(=O)ccn(C)c3)=O)C(C2)C1 CN1CCN(C)C(CNC(=O)C2=CCC(NC(c3cccc4cc[nH]c34)=O)C2)C1 N1(C(C2N(C(C)=O)C(=O)CC2)=O)CCN(C(c2sc(O)nc2C)=O)C2(CC2)C1 N1(C(c2ccnnc2)=O)CCC2CCC(C1)N2C(C1CCc2ccnn2C1)=O C12(NC(CCOc3ccc(C)cc3)=O)CCC(CC1NC(=O)C1=COCC1)C2 c1(C)nc(N(SC)CC2CCCCC2)cc(C)n1.C1(C)(C)CC=CCC1 CC1(C)CCN(C(C2Cc3nccn3C2)=O)CC1C(=O)NCc1cnsc1 c1(C(N2C(CNC(Cn3c(CCC)ncc3)=O)CC(O)C2)=O)c[nH]cc(Cl)c1=O c1(C(N(C)CC2CCCN(C(c3cnsn3)=O)C2)=O)ccc(F)cc1NC(N)=O c1(C(=O)NC(C)CCNC(=O)C(C)c2ccco2)ccc(N)cn1 N1(CC(C)C)CCC(NC(C2CCc3nncn3C2)=O)CC(C)(C)C1 CCC1=NOC(C(N2CCCC2(C)CCC(=O)N(C)Cc2ccnn2CC)=O)C1 N1(C(c2c(C)scc2)=O)CC2CCCC(NC(=O)Cn3ccc(C4CC4)n3)C2C1 c1(CNC(=O)NCc2ccc(C(F)(F)F)cc2)nc[nH]c1[N+](=O)[O-] C1(NC(c2c(C)nco2)=O)CCC2CN(C(=O)C(F)C(C)(F)F)CC12 N1(C(C(c2ccncc2)C)=O)CCC(OCCNC(c2c[nH]cc2C2CC2)=O)C1 C1(N(C(c2c(COC)nn[nH]2)=O)C)CCCN(C(C2CCCCC2(C)C)=O)CC1 C(CCN=c1[nH]nc(C(F)F)o1)NC(=O)C=C1CCCCCC1(F)F C(=O)(C(CC(F)F)c1ccccc1)NCCN(C(c1cccnc1SC)=O)CC CCC(CC(=O)N1C(C(=O)NCc2nnc(C)n2C)CCC12CC2)CC(C)C C1(CNC(=O)CC2C=CCC2)COCCN1C(C1CC=CCO1)=O N1(C(C2CC(NC(COCCCCC)=O)C2)=O)Cc2ccccc2C1 Cc1cc([N+](=O)[O-])ccc1C(=O)NN1C(C)CCCC1.c1(N)c([N+](=O)[O-])cnn1C C1(C(=O)NCC2CC(CC)C2)C(C)CCN1C(c1ccc(N)cn1)=O C(C(C)C(=O)NC(C)(C)C=CC(=O)NCc1n[nH]cc1C)OC(C)=O C(=O)(C(C)(O)C(F)(F)F)N(CC(CC)NC(c1cc(C)nc(O)c1)=O)C C(N=c1cc(C)[nH]c(=NCC23CCCC(CO2)C3)[nH]1)c1cc(OC)c(C)cc1 c1(CC(CCOC)NCC2CC(F)(F)CN2)cccc(Br)c1 Cc1nc(C)c(C(N2CCCC(NC(=O)C(C)ONC(=O)OC(C)(C)C)C2)=O)s1 Cc1ccc(F)c(C(N2CCC(C(C)(C)C(=O)NCC#CC(C)(C)C)C2)=O)c1 N1(C(C#C)=O)CCC(C2CCN(C(=O)CCOc3ccccc3CC)C2)CC1 c1(C(=O)NC2C(CNC(c3cc(C)sn3)=O)CCC2)cc2ccsc2s1 c1(C(C)NC(C(=O)N(CCCCC)C(C)C)=O)nnc(O)o1 N1(C(c2nc(CC)oc2C)=O)CC(CNC(=O)Cc2ccsc2)OC2(CCC2)C1 N1(C(c2cn(CC)nc2)=O)CC(NC(C2(C)C=CCC2)=O)C(O)C1 C(=O)(CC(C)(C)C(F)F)NC1(C(=O)NCCCOCC2CCC2)C(C)CCC1 C12(C(N3CC(O)(CCNC(C4C(C(N)=O)CC4)=O)C3)=O)CCCN1S(=O)(=O)CC2 C1(NC(CC2CC(CC)C2)=O)CC(C(=O)NCC2(Cl)CC2(F)F)=CC1O c1(-n2cc(C(N3CCC34CCC(C(F)F)CC4)=O)nn2)ccc2c(c1)OCCO2 N1(CCCNC(c2cnn(C)n2)=O)CCN(C(=O)C(O)Cn2cncn2)CC1 C1(CN(C)Cc2sccc2-n2cnnn2)CCCC(CNC(C2CC(C#N)C2)=O)C1 c1(C(C(C)NCC23CC(CC2CO)C3)OCC)ccc(F)cc1F c1(NC2CCCN(C(C(C)(C)C3CCCCC3)=O)CC2)ncc2ccsc2n1 C(=O)(C(CO)C(C)(C)C)NC1(CF)CCN(C(c2cccc(C#C)c2)=O)C1 C#CC1CC2(CC2)CN1C(C1CC(C)(C)CN1C(c1ccn(CCF)n1)=O)=O N1(C(CC2C(OCC)CC2)=O)CCC(O)(CNC(C2CCC23CCCO3)=O)CC1 O=C(C1CCCc2nncn21)N1CCC(CO)C(NC(C2(C(F)F)CCC2)=O)C1 N1(C(C(C)SCCCC)=O)CCc2[nH]nc(CNC(=O)C(C)OCOC)c2C1 C(c1ccc(F)c(F)c1)=CC(N1CC(CN(C(=O)C(C)(C)C#N)C)C2(C1)CC2)=O C(=O)(N=c1[nH]oc2cnccc12)C1C(NS(CCOC)(=O)=O)CCC1 c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(=Cc3cnc[nH]3)C)C2)c(F)c(Cl)c1 N1(C(CC(=C=C)C)=O)CCN(C(=O)C(c2ccc(Br)c(C)c2)C)CC1CC C1(OC)CC(NC(c2cn(C)c(=O)n2C)=O)CN(C(=O)CC2(C#N)CCC2)C1 Cc1nc(C2CCCC(C(F)F)C2)n(-c2ccnc(SC(C)C)c2)n1 C1(NC(c2ccc(OC(C)C)cn2)=O)CCC(C)N(C(c2ccc(F)s2)=O)C1 CC(CC(=O)NC1CN(C(C2CCn3c(cnc3C)C2)=O)CC1C)CC(C)(C)C c1(OC)ccc(OC)c(CC(=O)NCC(CO)NC(=O)CC(C)F)c1 c1(C(N(CCc2cn(CCN(CC)CC)nn2)C)=O)cc(C(C)C)nc(O)c1 Cc1cc(N)cnc1C(=O)NCc1cccc(C(=O)NC(C2CCCO2)CO)n1 C(N=C(NCC1(Cl)CCOCC1)N1CCC2(CCOC2)C1)c1ccc(F)cc1 CN1CCC(O)(C2(C(=O)N(CCCCN(C(=O)Cc3ccon3)C)C)CC2)CC1 c1(OC)nccc(I)c1C(N1CCOC(C(=O)Nc2ccc(Br)c(O)c2Br)C1)=O O=[N+]([O-])c1cc(Cl)c(S(=O)(=O)Nc2cnc3n2CCS3)c(Cl)c1 c1(C(N2CC(CC)N(C(=O)CN3CCC(F)(F)C3)CC2)=O)ccc(F)cc1C#N Cc1nsc(C)c1C(=O)OC1CC(=O)N(C)C1 C(C(CC)(CC)C(=O)NCCc1ccnc(C)n1)NC(C(C)NC(CC)=O)=O c1(CNC(N2CCC(COCCOC)C2)=O)ccc2c(c1)C(=O)CCS2 N1(C(C=CCC2(OC(C)C)CCC2)=O)CCC2(CCCCO2)C1.C1C(=O)N1 c1(CN(C(c2ccsc2OC)C(=O)NC(CC)C)C)ccc([N+](=O)[O-])cc1OC C(=O)(CCCCCC(C)C)NCCC(C(N1CCN(C)C(=O)C1)=O)OC C(=O)(CCC(=O)NCCNC(c1c(-c2cccc(F)c2)noc1C(C)C)=O)NC C(=O)(C(C)(C)COC)NCC(CC)NC(=O)OC(C)(C)C.C12(C)CCN(C1)C2=O c1(C(=O)NC2CCN(C(C(C)C(C)(C)O)=O)C2)ccc([N+](=O)[O-])c(C#N)c1 c1(C(=O)OC)cc(Cl)cnc1NC(C12CC1CN(C(c1cnc(C)cn1)=O)C2)=O C1(NC(Cc2nn(C)c(Cl)c2)=O)CCN(C(c2ccccc2C2CC2)=O)CC1F c1(CC(=O)NC2C=CCN(c3ncncc3Br)C2)cccc2sccc12 c1(OC(C)C(=O)NC2CN(C(c3cnns3)=O)CC2F)cccc(CO)c1 CC(CC(C)(C)CO)NC(=O)COC1CC(NC(c2ccc(Cl)s2)=O)C1 c1(C(=O)NCCC2(NC(CNC(=O)OC)=O)CCC2)nc(C)n(C)n1 N1(C2CN(C(C3C(C)CCN3)=O)C2)CCC(C#N)C1 C1(CC(=O)NC2C(NC(=O)CCCn3ccnc3)CC2)CC12CC2(F)F C1(CCC(=O)NCCC2CCCO2)CCN(C(C2CC(Cl)(Cl)C2)=O)CC1 C#CCC(C)(C)C(=O)NC1CN(C(=O)C(c2ccc(OC)c(F)c2)C)CCC1C C1(C(=O)NC(c2ccc(CNC(=O)C(c3ccccc3)F)cc2)C)C(C)(C)C1(F)F C1(C(=O)NC(CN(CC)CC)C)CCOCC1NCC.C(=O)(C(C)(O)CC)NC c1(C(=O)NC2C(C)CN(C(c3cccc(C(F)(F)F)c3)=O)C2)cccc(Cl)c1O N1(C(C=CCC)=O)CC2OCCN(C(=O)CCc3ccc(OC)nc3)C2C1 N1(C(c2cccc(OC)c2)=O)CC(NC(c2nc(C)nn2C)=O)C2(CC2)C1 C1(NC(C)=O)CCC2CN(C(c3ccc(C(c4[nH]nnc4C)=O)cc3C)=O)CC12 c1(C(N(C2CCC(NC(=O)COCCCF)C2)C)=O)cc2ccsc2c(O)n1 c1(CNC(=NCC=C)NC2CC(OC)C2)ccc2cc(F)ccc2c1 CC1CN(C(C2C(NC(=O)CCOC3CCCC3)CC2)=O)CC(=O)N1C c1(C(C)NC(c2nnnn2CCOCC(C)C)(CC2CC2)C)cocc1Br.CO c1(C(=O)O)ccc2c(C(N3CCC(N4CCOCC4)C3)=O)n[nH]c2c1 CC(F)(F)C(F)C(=O)NCC1(F)CCCN(C(=O)C(=C2CCCCC2)F)C1 CC1CCC(C)C1NC(=O)C(Cc1cnc[nH]1)NC(=O)C(=O)NC1CC1 C1(N(C(CC(CC)C)=O)C)CCCN(C(=O)CN(C2CCSC2)C)CC1 C=C(C)CC(C(=O)Nc1cccc(CCF)c1)NC(=O)CC1CC(C2CC2)C1 Cc1[nH]cc(C(N2CC(NC(C3(F)CC3)=O)C(N=[N+]=[N-])C2)=O)c(=O)c1Cl N1(C(c2n(CC)ncc2)=O)CCC=C(C(=O)NC2CCOC23CCCC3)C1 c1(CC)cc(C(N2CC3(CCC3NC(=O)CC(C)C3CCCC3)C2)=O)ccc1C S(=O)(=O)(c1ccc(F)cc1F)NC(c1ccccc1)C(=O)O c1(Sc2ccccc2)cccn(C)c1=O.c1(NC(C2CC2N)=O)cncc(CO)c1 C1(CNC(CSc2nc(C)[nH]n2)=O)CN(C(=O)Cc2ccns2)C(C)(C)C1 N=c1cc(C(N2CCC(O)(CNC(c3ccc(Cl)o3)=O)C2)=O)nc(Cl)[nH]1 C1(CNC(CC(=O)NCC)=O)CCN(C(c2cn(C)nc2-c2ccoc2)=O)CC1 C1(C(N2CC(n3cc(CNC(C4CCCCS4)=O)nn3)C2)=O)CNC(=O)C12CC2 CC(CCN(C)C)C(=O)N1CC2CC2C1C(=O)NCCc1cccc(F)c1 CC1(C)CCN(C(C2CCC(C)CC2)=O)CC1CNC(=O)C(F)F C1(CC=C(CC)C)CN(C(C2(CC3CCCCN3C(C)=O)CCC2)=O)CCO1 c1(OC)ccncc1C(=O)NCC(C)CNC(=O)C(F)(F)c1ccccc1 C1(C(N(CCCc2ccco2)C)=O)CCN(C(=O)CC2(C#N)CCC2)CC1O c1(OC)c(NC(C2CC(O)CN2C(c2occc2Br)=O)=O)ncnc1Cl C12(NC(C(CN(C)C)O)=O)CCC(C1)N(C(=O)CCc1ccc(O)c(Cl)c1)C2 Cc1ccc2c(c1Br)CCCN2C(c1ccc(F)cc1F)C(=O)NC1CCOC1 Cn1ccc(=O)c(C(N2CCC=CC2C(=O)NC2(CO)CCC2)=O)c1 CC(C)(C)CC(O)C(=O)NC1CN(C(c2ccnc3ccnn23)=O)CC1(C)C c1(C(=O)NCC23C(CN(C(C(CN(CC)CC)F)=O)C2)C3)cnc(O)cc1C C1(C(=O)NC2(CC(=O)NC(CC=C)C)CC2)CC(C#N)C1 c1(CC#N)ccc(C(=O)N(C2CCN(C(C3(C(F)(F)F)CC3)=O)C2)CCO)cc1 c1(CC(=O)NC2CC(CNC(C(c3ccc(Cl)cc3)CC)=O)C2)ccc(O)nc1 c1(C(N2CC3CN(C(C4N(CC)CC4)=O)C3CC2)=O)cc2nc(=O)ccn2[nH]1 CC(C)CC(C)(C)C(=O)NC(C)CCCC(=O)N(CC(F)F)CC(C)O c1(OCC(=O)NC(c2cn(C)nn2)c2ccccc2)ccc(C#N)cc1Cl C(C1=NOC2CN(C(c3c(C)nn(CC)c3C)=O)CC12)NC(C=CC=CCC)=O N1(C(C(C)(C)O)=O)CCOCC2(C1)CN(C(=O)Cc1cccs1)CCCO2 C#Cc1ccc(C(=O)NCC2(NC(=O)C(CCC)OC)CCC2)cc1F C1(CC(N2CC3(CC(NC(C(C)SCCCC)=O)C3)C2)=O)CCCC(C)(C)CC1 c1(C(=O)NCCOC)ncncc1OC.C1C(=O)N1CCCN(C)C c1(OCCCC(=O)NCC23C(CN(C(C4C(C=C)C4)=O)C2)C3)c(C)cccc1C C1(OC)CC2(C1)CN(C(=O)C(O)CNC(=O)C(C)C(F)(F)F)C2 N1(C(C(C)(C)CCCF)=O)CCCC2(CCC(NC(c3ccns3)=O)C2)C1 C(=O)(CCCS(C)(=O)=O)NCC1C(C)(C)CN(C(=O)Cn2cc([N+](=O)[O-])cn2)C1 N1(C(C=CC(C)=O)=O)CC2(C1)SCCC2NC(C1CC12CCSCC2)=O C1(C(=O)NC(CC(C)C)(C)CNC(C2COC(C)C2)=O)CN2CCCN1CC2 C(=O)(C(F)C(C)C(F)(F)F)NCC1C(C)CCN1C(=O)C=CC1CCOC1 C1(c2nnnn2CCCOC(C)(C)C)(NCC2(C)COC2)CCCC1C1CC1 CC(Cc1ccccn1)C(=O)N1CC(O)(CNC(=O)CCC2CCC(C(N)=O)O2)C1 c1(CNC(c2ccc(CNC(C(COC)(C)C)=O)o2)=O)cc(C)c(C)nn1 c1(C(N2CC(CCC)C(SC)C2)=O)cnc2cc(C)nn2c1 N1(C(C(n2cc(-c3c(C(=O)OC)cc(F)cc3)nn2)C)=O)CCC2(CC1)CSC2 c1(C(C(=O)NC2CC2)N(C2CCC(C)C2)CCOC)cc2cccc(Cl)c2s1 C1(CNC(COc2cn(C)nc2)=O)C2CCC(C2)N1C(C1(S(C)(=O)=O)CCC1)=O C#Cc1cccc(C(=O)NC(CNC(c2cc(C(C)(C)C)no2)=O)C(C)C)c1F C1(NC(C2C(C)CCCC2)=O)CN(C(c2ccn(C)n2)=O)CC(C)(C)C1 C1(C(=O)NCCC(=C)CNC(=O)CCc2cccnc2Cl)CCCN1N=O c1(N(CC(=O)NC2CC(NC(C=CC(C)OC3CC3(F)F)=O)C2)C)ccccc1 C(C)(C(C(C)C)NC(c1ccc(CO)o1)=O)NC(CNC(C)=O)=O c1(C(=O)NC(CNC(c2ncn(CC)n2)=O)(C)C2CC2)ccc2nnc(O)n2c1 CCC(C)CCCCC(=O)N(CCCNC(=O)C=Cc1cnccc1C)C c1(C(=O)NCCN(C(C(CC=C)C(C)C)=O)C)coc2c(C)cccc12 C(=O)(C(C)(O)C(C)(C)C)Nc1c(COC)cc(C(=O)O)cc1 Cc1nc(NC2CC(CNC(c3cnn(C)c3C3CC3)=O)C2)c(F)c(C)n1 CCCC(C(=O)OC)C(=O)N1CC2(CCN(C(=O)CC3CCCC(C)C3)C2)C1 Cc1cc(C=CC(N2CCCN(C(=O)C(C)CF)CC2CO)=O)ccc1Br NC(=O)C(CCC(=O)O)NCc1ccn(-c2cc(F)ccc2F)n1 Cc1cc2c(cc1-n1cc(CN(O)C(=O)CCC3(C#N)CCC(C)(C)C3)nn1)OCO2 N(C(=NCC1CCCC1)NCc1ncoc1C)CC(=C)C c1(C(=O)NCC2CN(CC(=O)OC(C)(C)C)C2)cc2cc(Br)cc(Br)c2o1 C1(NCC(=C)CCNC(=O)CC(=O)N(C)C)CC(=O)NC(c2cnn(C)c2)C1 CCC(CC(=O)NCC(C)CO)N(C(=O)CC1(C)OCCO1)C CC1C(C(=O)NCCS(N)(=O)=O)CCN1C(C1CC=CC1)=O C1(C(N2C(C(=O)NC3CCC(OCC)CC3)CCCC2)=O)CC(C)CC(C)C1 CCC1=NOC(C(=O)NC(Cc2ccccc2)CC(=O)Nc2cc(OC)ns2)C1 c1(C(=O)NC(C(C)NC(=O)COc2cncc(Cl)n2)CO)ccc(N)c(Cl)c1O N1(C(CC2(NC(C(C)n3cccc3)=O)CC2)=O)CC(O)C2(CCCC2)C1 N1(C(=O)C(Cl)=CCl)CCC2(C1)CN(C(c1ccc3nn[nH]c3n1)=O)CCO2 Cc1cnc(F)cc1C(C(=O)Nc1ccccc1Cl)N(C)Cc1cncn1C CC1(C)CCOC(CC(N2CCN(C(=O)Cc3ccc(F)nc3)C(CF)C2)=O)C1 Cc1cc(C(N2CCC(CO)C(NC(=O)CC(C)CN(C)C)C2)=O)cc(N)c1 CC1C(NC(=O)CN2CC3CC3C2)CCCN1C(c1ccc(CC2CC2)cc1)=O c1(CNC(C2CC(C)(NC(C(CC)C#N)=O)C2)=O)ccc2n[nH]cc2c1 C=CCCC(C=O)OCC.C12(NC(c3ccccc3)=O)CCCC1OCC2 C1(CNC(c2ccc(Br)cc2)C2CCOCC2)CCC2COCCC2C1 S(=O)(=O)(c1ccc(NCC2CC=CCC2)c(F)c1)N(CCCO)C C1(C(=O)NCC(C(C)C)NC(=O)C(F)C2CCC2)CC2CCCC(C1)C2 c1(C(N2C(C(C)OC)CCCC2)=O)[nH]c(=N)ccc1C.c12nocc1C(=O)NC2 c1(CC)csc(CCNC(c2nnnn2CC(F)F)NC(=O)OC(C)(C)C)n1 N1(C(Cc2c(C)nsc2)=O)CC(N(C(=O)C(C)C(F)(F)F)C)C(C)(C)C1 N1(C(CCCC=C)C)CCN(C(=O)N(CC(=O)OC)C2CC2)CC1C C12(NC(CNC(=O)NC)=O)CCCC1(C)CN(C(c1cccc(C)c1Br)=O)CC2 c1(C(N2CCC(NC(C3CC(C#N)(OC)C3)=O)C2)=O)cn2nc(C)cc2[nH]c1=O c1(CC)cc(Cl)ccc1C(N1CC(NC(c2cscc2OC)=O)C(C)(C)C1)=O C(CCCCC(=O)N1CCCC(C)(NC(c2nnc(O)cc2O)=O)C1)N(C)C C(=O)(C(F)CC(C)C)N(CCNC(CCCN(CCC#C)C)=O)CCC C1(CCC)(NC(c2cnco2)=O)CCCN(C(c2cccc(C(C)C)c2)=O)C1 N1(C(CSc2ccc(OC)cc2)=O)CCC(NC(=O)C(C)=C(C)C)C(C)C1 c1(C(=O)NC(C)CCCNC(=O)C#CC2(C)CC2)coc(S(N)(=O)=O)c1 C1(NC(c2c(C)nco2)=O)CN(C(c2cnn3c2OCC3)=O)CCC1CO N1(C(C2(C)C(C)(C)C2)=O)CCC2CCN(C(=O)CCc3ccc(O)nc3)CC2C1 CC(C)C(C(=O)N1CCCC(NC(c2cc(-c3ccccc3)co2)=O)C1)NC=O N1(C(CC(CC)N(C(C2CC2C(N)=O)=O)C)=O)CCC(=O)N(C)CC1 C(=O)(CC(=O)NCC(C)(Cn1cccn1)NC(C1CCCN1C)=O)NCC#C c1(CN2CCC(O)(C(=O)Nc3cnc(OC)nc3)C2)ccc(OC)c(Cl)c1 CCC(C)(CCNC(=O)CC1CC12CC2)NC(=O)C=Cc1cnn(C)c1 C(=O)(C1=CCCCC1)N1C(CC(=O)NCc2cnc(C)[nH]2)CCCC1 N1(C(C2N(C(c3ccc(C)o3)=O)C(C)C2)=O)CCCC2C(=O)OCC12 n1(CC(=O)N(C)CC2CN(C(=O)C(O)CC(F)(F)F)C2)c(O)nc2ccccc12 c1(C(=O)NCC(C(C)C)NC(C(CC)OC)=O)cccc(-n2cncn2)c1 Cc1cc(Cl)ncc1CC(N1CC2CC(CNC(=O)C(C)(C)N(C)C)C2C1)=O N1(C(CC=C(C)C)=O)CC2CC(C)N(C(c3ccn(C4CCC4)n3)=O)C2C1 C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cnc(N(C)C)o2)=O)C1 C=CCC(C)C(=O)N(C)CCOCCNC(=O)CC1CC2CCC1O2 Cc1csc(CCNC(=O)C(C2(O)CN(C(c3ocnc3C)=O)C2)F)n1 c1(C(N2CCC(C(C)NC(C3C(=C)CC3)=O)CC2)=O)csc2cccnc12 CCC(C(=O)NCCN(CCOC)C(C1CSCN1C(C)=O)=O)n1ccnc1 C(=O)(C1Cc2ccc(F)cc21)NCC#CCNC(c1cc(N)c(Cl)cc1)=O C1(NC(c2nc(C)[nH]n2)=O)CC(F)CN(C(=O)C(C)NC(=O)Cn2cnnn2)C1 C#CCCCC(C)C(=O)NC12CC(NC(=O)CCC(=O)OC)(C1)C2 c1(C(C)C)nc2[nH]ccc2c(=Nc2cccc(O)c2)[nH]1 c1(C(=O)NC2(COC)CCN(C(=O)Cc3cn[nH]c3)C2)cc2ccccc2o1 C1(CCN(C(C(C)CO)=O)C)CCCCN1C(=O)CCCOc1ccccc1Cl O=C1CC(C(=O)NCCC2(NC(c3ccc(Br)c(O)n3)=O)CCC2)=NN1 C(CCCCCNC(=O)CCF)N(C)C(c1cnoc1C1CCOCC1)=O C(C)(C)(CC(F)C(=O)N1CCC2CC12C)NC(C(CC)CC)=O C(C(C)(CC(C)C)NC(=O)C(C)OCCC1CC1)NC(Cn1nc(C)oc1=O)=O N#Cc1cnc(NC(C2CC2NC(=O)CC2CC2)=O)c(I)c1 C12(C(=O)NCCN(C(c3cccn3C)=O)CC)CCC(=O)C(F)(F)C1C2 C1(NC(c2cc(CNC(CCC(C)OC)=O)nn2C)=O)COCCC1(F)F N1(C(C(CC)N(C(CC(C(=C)C)OCC)=O)C)=O)CC2CCCC(O)C2C1 C1(C)(C(=O)NCC2CN(C(C3(CC#C)CC3)=O)CC2C)C(C)(C)C1(C)C C1(C(=O)NCC2CC3CCC2C3)(CC)CCN(C(c2nonc2N)=O)CC1 C(C)(C)(C(C)CC(=O)N(C(C)CS(C)=O)C)NC(c1c(CC)noc1)=O c1(C(N2C(Cc3cn(CCCC)nn3)CCC2)=O)cncc(-n2cccn2)n1 Cc1nc2cc(C(=O)NC3CC(N(C(=O)C(C)n4ccnc4)C)C3)[nH]c2s1 C1(CCC(=O)N(C2CCCCC2)C)CCCN(C(C23COCC2C3)=O)C1 Cc1c(C(N2CC(O)CC2CNC(=O)C(C)CC2CC2)=O)ccc2c1CCC2 N1(C(c2c(C)ocn2)=O)CC(C)CN(C(C2CC2C2CC2C)=O)C(C)C1 C1(C)(C(=O)NCC2CN(C(c3c(OC)scc3)=O)C(C)C2)CC2(CCC2)C1 C(C)(C(=O)NCCn1cnc(C(=O)NC(C)C(C)(C)C2CC2)c1)(C1CC1)OC N1(c2cc(C#N)ncn2)CCC2(CCCN(C(C3CNC(=O)O3)=O)C2)C1 C(=O)(C(F)CC(C)(C)NC(=O)CCC1CCOC1)NCc1c(C)nn[nH]1 Cc1ccc(NC(C2CCCN2C(=O)Cc2cccc(F)c2)=O)c(C)n1 C1(C(=O)NC(CN(C)C(C2CC(N(C)CCO)C2)=O)(C)C)CC(F)C(=O)N1 N1(S(CC)(=O)=O)CCC(C(=O)NC2CN(C(=O)CCc3cccc(O)c3)C2)CC1 C(=O)(CC(C)C(C)C)N1CC(CC(=O)NCCN(C(C)C)C)C(C)C1 C(N=c1nc2sccc2c(N2CCOC3(CC3)C2)[nH]1)C1C(=O)N2C1CCCC2 CCCCCCCCCCC(=O)NCC1CN(C(=O)CNC(C)=O)CC1(F)F c1(OC(C)C(=O)OCCOC(c2ccccc2F)C)ncc2ccccc2n1 c1(C(=O)OCC)nnc(SC)nc1N1CCCC1C(C)NC(C1CC(=O)N1)=O N1(C(c2cnc(C)o2)=O)CCC(C(=O)NCc2nc[nH]n2)CC1C C1(CNC(C(CCSC)O)=O)CCCCCN1C(=O)Cn1cccc(C)c1=O C1(C(=O)NCCC2(OC)CN(C(C(COC)(C)C)=O)C2)CC1C1CCCC1 c1(-c2nc(C)on2)ccc(CNC(=O)NC2CC=CCC2C)cc1 c1(C(C)C(=O)NC2CCN(C(C)C(=O)N(C(N)=O)C(C)C)C2)ccc2c(c1)OCO2 Cc1nc(N2CCC(CCC3CC3)CC2)c2c(C)c(C)sc2n1 c1(NCCCCCCCC=C)[nH]c(=NCc2cncn2C2CC2)nc2sccc12 CCN=c1[nH]cc(C(=O)NCCCCC(C)NC(c2cnn(C3CCOC3)n2)=O)s1 C(=O)(CCC(=O)NCC1(CCNC(c2[nH]c(C)nc2C)=O)CC1)OC c1(-c2nccc(CNC(=O)C(CO)Sc3ccccc3)c2)cncc2nc[nH]c12 CCC(C)C(CC(=O)NC(COC)CCO)NC(=O)CC1CCC(=O)NC1 N1(C(C2(CC)CCC2)=O)CCC2CC2(C(=O)Nc2ccc(CCF)cc2)CC1 Cn1nc(Cl)c(C(=O)NC2CCCCN(C(c3ccc(CO)c(Cl)c3)=O)C2)c1Cl C1(C(=O)NC(c2ccccc2F)CNC(CC2CC(=C)C2)=O)CCN(C)C1=O C1(NC(c2cccc(C(F)F)c2)=O)CN(C(=O)CCC2CC2(F)F)C2CC12 c1(CNC(=O)C(C2(O)CCCC2)F)c(C(=O)OC(C)(C)C)nc2n1CCCC2 c1(NCC2(C#N)CC2)cccn2ncnc12.N1CC(C=O)CC(F)C1 c1(N2C(C)CC(NC(c3cnn[nH]3)=O)CC2)ncc2ncn(C)c2n1 C1(NC(c2n[nH]c(C)c2F)=O)CCN(C(c2ccnc(F)c2N)=O)C12CCC2 c1(C(N2CC(CCC)C(NC(=O)C(C3CC3)OC)C2)=O)cc(F)c(F)c(N)c1Cl C#CC1(C(=O)NC2CCCCC2NC(c2cc[nH]c(=N)c2)=O)CCCC1 c1(C(N(C2CCCC(NC(CNC(=O)OCC)=O)C2)C)=O)nn(C)c(=O)cc1C c1(C(=O)NCC(CC=C)NC(=O)CCCc2ccc(Br)s2)ncccc1C C1(NC(c2nc(CCCC)sc2)=O)(CC)CCN(C(=O)COC(F)(F)F)CC1 N1(C(CC2(COC)CC2)=O)CCCC12CCN(C(=O)C(n1cc(Cl)cn1)C)C2 N1(C(c2ccc(OC)c(C)n2)C(=O)NC)CC2(CCOCC2)c2ccccc21 Cc1ncc([N+](=O)[O-])cc1N(C1CC2CC1CN2)C(c1ccc(F)nc1C)=O C(CCN(C)C(c1ccc(O)nc1Cl)=O)(C(C)(C)C)NC(C(CC)NC(C)=O)=O C(C(C)(C)CNC(=O)CCN1CCC1)N(C)C(C1(N2CCCC2)CCC1)=O C1(C(N2C(C)(C)C(CNC(c3cnsn3)=O)CC2)=O)Cc2ccc(F)cc2O1 C(=O)(C#CC(C)(C)CNC(C1CCOC1)=O)Nc1c(C)ccc(O)c1 c1(CNC(N(C(Cc2cccnc2)CO)C)=O)nc(-c2ccccc2)cc(O)n1 C1(NC(c2cc(C)c(F)cn2)=O)CN(C(C2(n3cccn3)CC2)=O)C2(CCC2)C1 C12(CNC(C(C)N(C)C)=O)CN(C(c3cc(C(F)(F)F)cs3)=O)CC(F)(C1)C2 N1(C(C2(C)CC=CCC2)=O)CC(C2CC2C(=O)NC2CCCSCC2)C1 C=C=CCC(=O)NCC(O)CNC(=O)CCC1CCOC1 N(C1C(=O)Nc2cccnc21)C(c1cc(F)ccc1I)=O c1(NC2CCC(N(C(c3cnc(C)n3C)=O)C)CC2)nc2ccc(O)cc2s1 N1(C(CCNC(C)=O)=O)CC2CCC(C1)N(C(c1cc([N+](=O)[O-])cs1)=O)C2 N=c1ccc(C(=O)NCC2CC2CNC(=O)C=Cc2ccsc2)c[nH]1 CC1COCCN1CCNC(=O)CC(C1CC1)NC(=O)CC1CSCCO1 C(C)(C(=O)N(CCC(=O)N1CC(C(C)C)C1)C(C)C)(C1CC1)OC N1(CCOC)CCC(NC(CC2CCCC2)C(=O)O)C1 c1(C(N2CCCC(NC(C3(COC)C=CCC3)=O)C2)=O)cc(F)ccc1C(F)F Cc1c(CNC(=O)NC2(C(n3ccnc3)C3CC3)CC2)csc1Br C1(C(=O)NCC(=C)CCNC(=O)CCc2ccccc2)CC2(CO1)CC(F)(F)C2 C12(C(N3C(CC)C=CC3)=O)COCC1CN(CCc1ccsc1)C2 c1(N2CCC(C)C2)ccc(S(=O)(=O)N2CCC(CC3CCCO3)C2)cc1Cl C1(CNC(CN(CC)CC)=O)CCC(C)N(C(c2ccnc(C(N)=O)c2)=O)C1 N1(C(c2n(C)cc(NCCNc3c(SCC)cccc3)n2)=O)CCC(=O)C(C)C1 C1(CC(=O)N(CCCC(=O)OC)C)CN(C(C2CCCCO2)=O)CC1C Cc1nccc(C(C)NC(C2CC2C(=O)Nc2cccc(O)n2)=O)n1 O=C(C#CC1CCCCC1)N1CC2CCCC(C1)N2C(C1CC2(CCC2O)C1)=O C1(CNC(CCn2c(C)ncc2)=O)C(O)C(O)CN1C(=O)Cn1ccc(C(F)F)n1 C12(NC(CCC)=O)CCCC1CN(C(c1cc(-c3ccccc3Cl)[nH]n1)=O)C2 C1(CC)CC(C(=O)NCC2CN(C(C3CCC(=O)O3)=O)CCN2C)CC(=O)N1 C(=O)(C1=NN2CCCN=C2N1)NCC(C(C)(C)C)NC(C1N(C)C(=O)NC1)=O N1(C(CCC2C(C)=NNC2=O)=O)CCOCC(F)(CNC(c2cocn2)=O)C1 N1(C(C2(C#N)C(C)C2)=O)CC2CCC1C(NC(=O)CNC(=O)CC(F)(F)F)C2 C=CC1CN(C(=O)Cc2csc(COC)n2)CC1N(C(=O)C(F)(F)CC)CC Cn1[nH]c(C(N2CCC(CCNC(=O)CSc3cccc(F)c3)CC2)=O)nc1=O S(=O)(=O)(C1CC1c1ccccc1)N(CC(C)C)CCCCl CCCC(CCC)C(=O)NCCCCCC(=O)NCc1ccc(F)cc1O C(=O)(C1=CC2CC=CCC12)NC1CC(NC(c2c(O)ccc(C(C)C)c2)=O)C1 c1(C(=O)NCC(C)CNC(=O)CCc2ccc(Cl)cc2)cccc2c1nnn2C N1(C(C(COC)O)=O)CCN(C(c2cc(O)nc(Br)c2)=O)C(CO)C1 N(C(=NCCF)NCC1CCOC(C)C1)CC1(COC)CCOCC1 CS(=O)(=O)c1cnn(CC(=O)NCC2(C)CC(NC(C3(F)CCCOC3)=O)C2)c1 C1(CN(C(N2CC(C)(C(F)(F)F)C2)=O)CC2CCCCC2)CC2(CCC2)C1 c1(SC)cc(C(=O)NC(C2CN(C(C3CC3(Cl)Cl)=O)C2)C)co1 C1(C(=O)NC2CCN(C(c3cn(C)nc3Br)=O)C2)CCn2c(O)nnc2C1 c1(OC)[nH]ccc1CNC(=O)C(C)N(C(=O)C(C)(F)c1ccon1)C N1(C(C(=O)NCCOCCCC)=O)CCC(NC(C2(C)CC2(C)C)=O)C(O)C1 N1(C(CC(C(C)C)C)=O)CCC(C2CCCN(C(c3c(N)cnn3C)=O)C2)C1 CC1CCN(C(=O)C=Cc2ccc(Br)s2)CC1CNC(=O)C1=CCC1 N1(C(C(C)CC2CCCC2)=O)CC(F)(F)CC1(C)CNC(c1cnn(C)c1)=O CC1(C)CC(C(N2CCC(O)C(C)(C)C2)=O)CN(C(=O)C2=CCCOC2)C1 C12(C(N3C(CN(C(=O)CN4CCCNC4=O)C)CCC3)=O)CCCC(C1)OC2 c1(C(=O)NCC(CN(C)C(c2cnoc2-c2cccs2)=O)O)nc(=O)n(C)[nH]1 C1(C(N2CCC(C(C)NC(=O)CC3CC3(C)C)CC2)=O)(COCC)CCOCC1 c1(C(=O)OC)oc2ccc(S(=O)(=O)NC(c3ccccc3)CN)cc2c1C CC1CCc2nc(C(N3CCC(OCCNC(=O)CCCC#N)C3)=O)ccc2C1 Nc1cccc(F)c1C(N1CCCC1CNC(=O)Cc1c(F)cccc1F)=O c1cc(C2(C3CCOC3)CC2)c2c(c1)COCCC2 c1(SC)ccc(C(=O)NC2C=CCN(c3ncc4c(n3)COC4)C2)cc1[N+](=O)[O-] CCC(C)CCC(=O)N1CCCCC1CN(C(=O)Cn1cc(CN(C)C)nn1)C CC1COC(C)(C)CN1C(C1CCCCN(C(C2CCSC2)=O)C1)=O Cc1cc(C(=O)NC(C(=O)NCc2ncoc2C)c2ccco2)co1 CCC(CC(=O)N1CCCC1(C)CCC(=O)NCCC(C)(O)C1CC1)SC C1(C(=O)NCCC2(OC)CN(C(=O)Cc3ncccc3C)C2)CCC(O)CN1C N1(C(COCCOC)=O)CCC(C(=O)NCc2ncc(C)s2)C1C Cc1cc(CC(N2CCC2(C)C(N2CCOCC2C(c2ncc[nH]2)=O)=O)=O)nn1C C1(N(c2nc(C3CCC3)no2)C)CCS(=O)(=O)C1.C1C(=O)O1 C1(CCOC)(NC(c2sc(F)cc2C)=O)CCN(C(C2(N(C)C)CC2)=O)CC1 c1(C(=O)NCC(CNC(c2ccc(C#C)o2)=O)O)cnc2sccc2c1 c1(C(C)C(=O)NCC2CN(C(C3(C)CNC(=O)C3)=O)C2)cc(Br)ccc1F Cc1ccnc(CNC(=O)C(C)N(C(c2ccncn2)=O)C2CC2)n1 C12CC(C)CN(C1)C2=O.C1(CC(=O)NCCC2(COC)CC2)CC(F)C1 CCC(C)(CCNC(c1ccc(C#N)o1)=O)NC(C1CCC(C)(C)C1)=O c1(OCC)nc(N2CC(C(=O)Nc3ccc(C)nc3C)C2)ncc1OC CC(C)C(C)(Cc1ccccc1)C(=O)NCCC1CCN(C(C2(C)CSC2)=O)C1 C1(c2cn(CC(c3ccccc3)NC(C(C)OC)=O)nn2)CCC(=O)CC1 O=C(NNc1c(F)cccc1F)c1ccc2ncccc2c1Cl c1(C(=O)NCC2CCC(NC(CCC(=C)C)=O)C2)cc2cc(OC)ccc2[nH]1 C(=O)(CCN(OC)C(=O)Cc1n[nH]c(C)n1)NCCCOCCOC c1(C(=O)NCC(CCNC(=O)C=Cc2ncc[nH]2)O)cc2ccccc2nc1O c1(-c2ccc(CCCCNC(CN(CC(N)=O)C3CC3)=O)o2)ccccc1Cl N1(CC(CO[Si](C(C)(C)C)(C)C)O)CCc2c(OCC(F)(F)F)cccc2C1 C(CNC(C1(Cl)CC1(F)F)=O)(C(=O)N(C)C(c1cccs1)C)OC CC1=C(C(=O)NC2CC(C)N(C(=O)CCN3CCCCCC3)C2)CCO1 c1(OC)cccn2ncc(C(=O)NCCCOc3ccc4ncsc4c3)c12 C1(CC(C)NC(c2occc2C2CC2)=O)CCN(C(c2coc(C#N)c2)=O)CC1 c1(C(=O)NCC2(F)CC(CNC(COCCOCC)=O)C2)cc(C)c(CC)cn1 C1(OC)CC(C(N2CC(C)(NC(=O)CCSc3ccc(C)cc3)C2)=O)CC1OC c1(C(=O)NCC2CCCC2NC(c2cocn2)=O)ccc(F)c(C2CC2)c1 C1(COC)(NC(=O)Cc2ccns2)CCN(C(=O)COCCCN=[N+]=[N-])C1 Nc1ncc(Br)nc1C(=O)NCC1CCC1NC(=O)C=C1CCOCC1 C1(CCNC(N(CC(C)C#N)CC2CCC(C)(C)C2)=O)OCCCC1(C)C c1(-n2c(CNC(CC(=C)Cl)C)ncn2)ccc2c(c1)OCO2 CCCC(C)(CC)C(=O)N1CC(CNC(C2(C#N)CC2(C)C)=O)C(C)C1 Cc1ccc2cc(C(N3CC4CC3C4CNC(=O)C=CBr)=O)oc2c1 C(=O)(C1=CCCOC1)NCC(C(=O)NC(C(C)C)C)CC1CCCC1 n1(CCOC)nccc1C(=O)NCC(O)CN(C(=O)CCCC1CCCC1)C c1(C(N2CC(CCNC(COCCC)=O)OC(C)C2)=O)ccc2oc(S)nc2c1 C1(NC(C2CCN(C(C)=O)CC2)=O)CN(C(c2csnn2)=O)C(C)(C)C1 c1(C(=O)OCC2C(NC(=O)OC(C)(C)C)CCC2)cnc2sccn12 C1(NC(C2(CCC)CC2)=O)CCCN(c2cc(Cl)c(O)nn2)C1C c1(OCC)ncccc1C(=O)NC1CN(C(C2CCC(F)(F)C2)=O)CC2CC12 CC1(C)CCCN(C(=O)CCNC(N)=O)C1CNC(c1cncc(Cl)n1)=O c1(COC(C)C(=O)NCc2cn(C3CN(C(=O)CNC=O)C3)nn2)ccccc1 N1(Cc2cccc(-c3nc(C)sc3)c2)CCC2(CCC3ON=C23)C1 C1(NC(c2cc(COC)no2)=O)CC2CCC1(Nc1ccnc(C(=O)OC)n1)C2 C(=O)(C1CN(CCSn2nccn2)Cc2ccccc21)OCC C1(C(C)(C)C)(CNC(=O)Cc2nc[nH]n2)CCN(C(c2cc(CCO)on2)=O)C1 C1(NC(CSCC)=O)CCC2CN(C(c3[nH]ccc3-c3ccccc3)=O)CC2C1 C(CC(C)C(=O)NCC1CCN(C(c2c(Br)nnn2C)=O)C1)OC C1(NC(CC2(C(=C)F)CCC2)=O)COC2(C1)CN(C(=O)CCSCCCC)C2 c1(N2CCCC(OC(C)C)C2)nc2ccccc2c(=NC(C)C2CCC2)[nH]1.C1(C)CC1 C1(NC(c2cc(CC)n(C)n2)=O)COC2(CNC(C3CC3F)=O)CC1C2 C(=O)(CCCC(F)(F)CO)N(CCC(C)NC(c1ccnc(Cl)c1O)=O)C c1(OC)cc(N)ccc1C(N1CCC(C(=O)NC2C3CC4C(C3)C24)C(C)C1)=O Cc1cc(NC(=O)Cc2ccco2)ccc1NC(=O)C=Cc1ncccc1C CC(C(C)C(=O)N1CCCC(CN(C)C(c2c(Cl)ccnc2Cl)=O)C1)S(C)(=O)=O C1(CC)CN(C(=O)CCOC2CCCC2)CCC1NC(=O)CC(C1CC1)C1CC1 Cc1nncc(C(N2CCCC2CN(C(=O)C=CSCc2ccco2)C)=O)c1C N1(C(c2scnc2Cl)C(=O)NCCCCCC)CCC2(CC=CCO2)CC1 N1(C(C2(COC)CCCO2)=O)CC(CNC(=O)C(O)Cn2cncn2)C(O)C1 c1(C(=O)OC)ccc(CCCC(=O)N2CCCC2Cc2cnn(C)c2)cc1F C(=O)(C1=CCCC1C)NC(CSCC)C(=O)NCCCCCCN(C)C C1(CNC(CCC=C)=O)CN(C(=O)C(C)SCCCC)CCC12CCC2 c1(CS(C(CC(CC)NC(C)(C)CC)C)(=O)=O)cc(OC)ccc1F CCCCC(C(=O)N(C1CCN(CC)C1)C)NC(=O)CSC c1(OC)ncccc1CC(=O)NC1CN(C(=O)C=CCN(C)C)CC1C(F)(F)F C1(C(=O)NCC2(C(=O)OCC)CC2)CC(C)N1C(=O)C=C(CC)CC Cc1cc(N2CC3CCN(C(c4ccc(F)nc4F)=O)C3C2)n2nc(C)cc2n1 c1(COC)nc(N2CCC23CN(C(c2ccc(C)c(I)c2)=O)C3)cc(O)n1 C(=O)(CC(CNC(C1(C)CCCCO1)=O)C1CCC1)NCCC(C)F c1(C2C(C(C(=O)NC3CC(O)(CNC(C4CCOCC4)=O)C3)O)C2)cccnc1Cl C1(N(C(C(C)OCCC=C)=O)C)CN(C(c2cn(C(C)C)nc2C)=O)CC1(C)C Cc1ccc(C(=O)N(C2CCCC2)CCCNC(=O)C2=NOCC2)c(Cl)c1C C=C=CCCC(=O)NC(c1noc(CC)n1)C C1(NC(=O)C(C2(O)CN(C(C3CC4CCC4C3)=O)C2)F)CCc2nncn2C1 C(=O)(CCCc1nncn1C)NCC(n1cc(C(C2CC2)C2CC2)nn1)C c1(C(=O)NC(C(=O)NCCNC(N)=O)CC(F)F)cc2cccnc2[nH]1 c1(CNC(C2C(C#N)C2)=O)cn(C2CN(C(=O)Cc3csc(C(F)F)n3)C2)nn1 C(=O)(C1COc2ccc(Cl)cc21)N1C2CC(NC(C=CC)=O)C1CC2 C1(C(=O)OCC)CN(C(=O)C2=NOC(C3(O)COC3)C2)CC12CCN2 c1(CC)c(C(=O)NCC2CN(C(=O)CC3CCC3)CCC2C)sc2ccccc12 c1(OCC)ccncc1NC(N1CCC(C(=O)Nc2ccccc2)C1)=O c1(NC(C(c2cccc(OC)c2)C)=O)cc(C(=O)O)c(C)c(C)c1 c1(N(C)CCC2CCCC2)nc(=NC2CC3(CCC3)C2)[nH]c2c1SCC2 C1(NC(C=CC(C)NC(c2n(CC)ncc2)=O)=O)CCCOC12CCC2 c1(N(C(CN2CCC(CC=C)CC2)=O)OC(=O)C2CC2)cnn2cc(Br)ccc12 C(=O)(C1=CNC2=NCCCN12)N1CCC(CNC(C(C)(O)C2CC2)=O)C1 C1(CNC(C2(CC#C)CCCO2)=O)CCN(C(=O)CCCC2CCC2)CC1O c12ccccc1CC(=O)NC(C)C(C)c1cn-2nn1.CC.OC c1(C(=O)NCC=CCNC(Cc2cc(C)nn2C)=O)cc(Cl)c(Cl)cc1C C(=O)(C1COc2ccccc21)NC1C(C)(CN(C(C=CC=CC)=O)C)CCC1 C1(C(N(CC(N2CCN(C(C(=O)NCC)=O)CC2)=O)C2CC2)=O)C2C(=O)OCC12Br.C C(C(C)(C)CC(=O)N1CCCCCC1CNC(=O)CCCC(C)=O)OC c1(C(N2C(CN(C(COCC(=C)C)=O)C)CCC2)=O)cccc(C#N)c1 C12(NC(C(CCC)OC)=O)CCC(C(=O)NCCc3ccncn3)(CC1)C2 c1(C(N2C(C)(C(N3CC(CC(=O)OC)C3)=O)CC2)=O)ccc(C)cn1 N1(C(CC(=C=C)C)=O)CC(F)(F)CC1CCNC(c1c(C)ccn1C)=O c1(SCCCC)cccc(C(=O)NC2CCN(C(C3CC34CCCC4)=O)C2C)c1 CCC(CCC(=O)N1CCCCC(NC(CC(=O)N(C)C)=O)C1)CCC(=O)OC CC(C)CC(C)C(=O)NC(CN=[N+]=[N-])C(=O)NCc1cncc(O)c1 c1(NC2(C)CC(C(=O)NC(c3cc(C(N)=O)[nH]n3)=O)C2)cnc(CC2CC2)nc1 Cc1cnc(C)c(NC(C2CCCC(NC(c3ccnc(O)c3)=O)C2)=O)n1 n1(CCNC(C=CC(C)C)=O)cc(C(=O)N(C(C)C)CC2COCCO2)cn1 N1(C(c2c(C)cncn2)=O)CCC2C(CCCN2C(=O)CN(C)C)C1 c1(CC)occ(C)c1C(N1CC(c2cn(Cc3occc3C(=O)O)nn2)C1)=O C(CC(C)C)(C(=O)OCC1CC1c1ccncc1)ONC(=O)C1C(OC(C)=O)C1 N1(CC(=O)NCC2C(NC(c3ccc(C)s3)=O)C2)CCCCCCC1=O C(F)(F)(C(F)(F)F)c1scc(SCC(=O)NC2CC2NC(=O)Cn2cnnn2)c1 C1(C(C(C)C)NC(CCn2ncc(C)c2)=O)CCN(C(=O)CCCC2CC2)CC1 c1(C(C(=O)NCCCCCN(C(=O)Cn2ncn(C)c2=O)C)O)ccc(F)cc1 C12CCCN(C1)C(=O)CCC(=O)NC2.C(C(=O)N(CC)CC)SCC#C c1(N(C(c2ccn(C(C)C)n2)C(=O)NCC2CCCO2)CC=C)cccc(Cl)c1 C1(CNC(CC(=O)NCC#C)=O)CC2(CCN(c3nc(CC)nc(=N)[nH]3)C2)CO1 C1(C)(CC)CC(NC(=O)C=Cc2ccsc2)CN1C(C1(c2cccs2)CC1)=O S(=O)(=O)(c1cc(C(=O)NC2CC3CC(NC(=O)CSC(F)F)C2C3)co1)NC CC1CN(C(c2c(Cl)cncc2Cl)=O)CCCN1C(c1cn(C)nn1)=O Nc1cccc(CC(N2CC(NC(=O)C=Cc3ccc(Cl)cc3)C2)=O)c1N c1(NCC2(O)CC(OCC)C2(C)C)cc(Br)cc2cn[nH]c12 Cc1cc(C(=O)OC(CCNC(=O)OC(C)(C)C)C)nn1-c1cccc(Br)c1 C(=O)(C(S(C)(=O)=O)C1CC1)NC12C(CN(C(Cc3nc(C)oc3)=O)C1)C2 c1(N(CCCC(=O)NC)C)ncccc1S(=O)(=O)NC(C)C(C)C(F)(F)F N1(C(c2c(COC)nn[nH]2)=O)CCC(C2CC2)C1CNC(=O)CC1(COC)CC1 C1(C(=O)NC2CN(C(C=CSC)=O)C2)CC(O)CN1C(C)=O N1(C(c2cc(C)c(F)cc2)=O)CCCN(C(=O)CCc2ccccc2O)C(C)C1 C(=O)(CC(C)CC(=O)N1CC(C(=O)NCCCOCC2CC2)C(CC)C1)OC CCCCC(F)C(=O)N1CCCC(C(=O)NCc2coc(C)n2)C1 C1(C(=O)NC2(CC#C)CC2)(NC(C2(CC)CCC2)=O)CCC(C)(C)C1 CN1C(=O)CSC1=CC(=O)NCC1CCN(C(C2COC3(CCC3)C2)=O)C1 C1(C(NOC(C)(C)C)=O)C(O)C(O)CN1Cc1c[nH]nc1-c1ccc(F)cc1C c1(Cc2cnn(C)c2N2CCOC(C(F)(F)F)(C(F)(F)F)C2)cn2ccsc2n1 Cc1ccnc(C)c1C(N1CCCN(C(=O)CCn2cncn2)CC1)=O C(=O)(CC(O)CN(C)C)N(CCN(C(c1cnc(C(C)OC)s1)=O)CC)CC c1(C(=O)NC(CN(C(=O)C(CCO)N(C)C)CC)C)ccnc(CO)c1 C(=O)(C(O)C(C)C)NCCC1CCN(C(C2C(C(=O)OC)C2)=O)C1 Cc1nc(C)c(C(N2CC(NC(c3sccc3-n3cnnn3)=O)C(C)C2)=O)[nH]1 Cc1ccc(C(C)CC(=O)N2CC(NC(=O)CCCc3ccc(C)cc3)C2)cc1 C(CN=[N+]=[N-])(C(=O)NCCN1CC=CCC1)NC(C1CCN(CC)C1)=O c1(C(=O)NC(C2(O)CCN(C(=O)Cc3cnn(C)c3)C2)C)cnc(O)cc1O c1(OC(C(=O)NCC(CO)OC)C(=O)OC)cc(Cl)cc(Cl)c1 c1(CC(=O)NC2C3CN(C(c4nc(CCC)sc4)=O)C2C3)ccc([N+](=O)[O-])cc1 C1(NC(c2ccn(CC)n2)=O)CN(C(=O)C(C)(C)Oc2ccc(F)cc2)CC1C C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC1C(NC(C2(C)CC(C)C2)=O)CCOC1 N1(S(CC(C)C)(=O)=O)CCC2(CCCC2C(=O)NC2CN3CCC2CC3)C1 C(C(O)CC(=O)NCC1(F)CCC(NC(c2csc(Cl)c2)=O)C1)N(C)C C1(N(CC#C)C(C2(C)CC2=C)=O)CCN(C(=O)CCN(CC)CC)CC1 C1(C2CCCN(C(=O)Cc3sc(C)cc3C)C2)(NC(CCC=C=C)=O)CC1 CN1CCCC(O)(CC(=O)NCC2CC(F)(CNC(c3cscn3)=O)C2)C1 c1(CN2CC(CNC(=O)Cc3cccc(Cl)c3)OCC2)ccc(O)c(Cl)c1 n1(CC)nc(C(N2CC(CNC(=O)Cn3cncn3)C(C)C2)=O)cc1C C1(NC(C2C(C)(C(F)(F)F)C2)=O)CC2CC(NC(=O)CN3CCCNC3=O)CC12 O=C(CC1=CCOCC1)NCC1CCC(NC(c2ccc[nH]2)=O)C1 C1(NC(CC=CC)=O)CC(C)N(C(C2CN(S(C)(=O)=O)C2)=O)C1 C(CC(C)(C)C)(c1n(CC(=C)C)nnn1)NCc1c(Cl)cnn1C CCC(CN(C)C)CC(=O)N1CCCCC(NC(c2cnc(O)n2C)=O)C1 n1(CC)cnc2c(NCC3(C4CC4)CC3)[nH]c(=NCCC(C)F)nc12 c1(CC)ccc(C(=O)NCC2(CNC(=O)CSC3CC3)CC(F)(F)C2)cc1 Cc1ccc2c(c1)N(C(C1CCCN(C(=O)CCn3nccc3C)CC1)=O)CC2 C(=O)(C1CCCc2ccccc21)NC1CC(CNC(C2(C#N)CC2)=O)CC1O c1(CCC(=O)NC2CN(C(c3c(C)cc[nH]3)=O)C3C2C3)cccc(Cl)c1Cl N1(C(c2c(C#N)csc2)=O)CCC2CN(C(=O)CC3CC(=O)NC(=O)C3)C2C1 c1(C(=O)NCCC(CNC(C(CC(C)C)OC)=O)(C)C)occ2c1CCOC2 C1(CC(N2CCCC(n3ccnn3)C2)=O)CCNC2(CCC2)C1 N=c1[nH]c(C(N2CCC(CNC(c3cnc(C4(N)CC4)o3)=O)C2)=O)cs1.C1CC1 Cc1cnc2cc(C(N3CC(N(C(=O)Cc4ccc(CO)cc4)C)C3)=O)ccn12 C1(NC(CSCCOC)=O)(CF)CCN(C(=O)C(=Cc2cnn(C)c2)C)C1 Cc1cc(C2CC2)ncc1C(=O)NCC1CCN1C(c1cc[nH]c1C1CC1)=O C(=O)(C(CNC(c1[nH]nnc1C)=O)C(C)C)NC(CC(=O)OC)(C)C CC1CN(C(C2CCC(C)C2)=O)CC1NC(=O)C(c1ccccn1)O Cc1cccc(CNC(N2CC(CNC(c3n[nH]cc3Cl)=O)CC2C)=O)c1 C(=O)(C1=CC2(CCOC2)C1)N(CCN(C)C)CC.C12CCOCC1NC2=O C(c1ccc(Cl)cc1)=CCc1cc(NC2C(O)CCC2)ncn1 c1(C(N(C)CC2N(C(CC(=C)C)=O)CCC2)=O)cccc2cccc(OC)c12 N1(C(C(=O)NC(c2onc(C)n2)C)=O)CCc2cc(Br)ccc2C1 CC1=NN(C)C(=O)C1CC(=O)NC(C)CCNC(=O)CCc1ccncc1 c1(C(N2CC(N(C(C3(F)C(C)OCC3)=O)C)C(C)(C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C=CC(C)(C)CC(=O)NC1CC(CNC(c2nc(Cl)sc2Cl)=O)C(O)C1 c1(N(S(=O)(=O)CC2CCN(S(C)(=O)=O)CC2)C)ccc(CCO)cc1 c1(C(=O)NC(CN(C(c2ccc(OC)s2)=O)C)C)cc2c(F)cc(F)cc2o1 c1(C(N2CC(NC(=O)CN3C(=O)CCC3=O)C3C2C3)=O)nccc2cccnc12 Cn1ccc2cc(C(N3CCC4(COC(CNC(=O)CO)C4)C3)=O)cnc12 c1(C(C)OC)ccccc1C(=O)Nc1ccc(CN2CCCC(C)C2)cc1 C(=O)(C(C)CC(C)C(C)=O)OCC.C1(N(CC)CC)CCN(C(C2(CCC)CC2)=O)C1 n1(CC)cnnc1C(=O)NCC(C)CNC(=O)C1=CCC1 Cn1cc(Cl)cc1C(=O)NC1(CCNC(=O)CC2CCCC2O)CC1 CCCC(C(=O)N(CCC)CCNC(c1coc(C(F)F)c1)=O)C(C)C CC(C)CC(C)(C)C(=O)NC1CCN(C(=O)C(C)(C)Br)CCC1CO c1(OC)ccccc1SCC(=O)NC1CCC(N(C(=O)C2=COCC2)C)C1 C1(OC)CN(N(CCF)CCC(F)F)CC1COC c1(C(=O)NCC(CNC(C2C(C)(C)C2(C)C)=O)OC)cc(Cl)cc(C)c1O N1(C(CC(C)NC(N)=O)=O)CC2(COC(CNC(c3cc4n(c3)CCC4)=O)C2)C1 c1(COC)ccc(C(N2CSCC2C(=O)NOCC2CCCO2)=O)o1 C1(NC(C(C)NC=O)=O)C2CCC1CN(C(c1cc3c([nH]1)CCOC3)=O)C2 O=C(NNc1c(Cl)cc([N+](=O)[O-])cc1Cl)c1c[nH]c2cc(Br)ccc12 C1(C(N(CCC(=O)NC)C)=O)CCCC1CNC(=O)CCCn1ccnc1 c1(CC(N2CC(C)N(C(C3(CO)CCCO3)=O)CC2)=O)ccc2c(c1)COCC2 N1(C(C(CC#C)(C)CC)=O)CCC(C2CC2NC(c2nncn2C2CC2)=O)CC1 C(=O)(C(F)C(C)CN(C(=O)CNC(C)(C)C)CC)N(CC#C)CCO C(CC1=CCCCC1)NC(CCC1CCC(NC(C(C)(C)Cl)=O)C1)=O c1(C(N2CCC(NC(C34CC(C)(C3)C4)=O)C(O)C2)=O)cc(O)c(F)cc1N C1(C(=O)OC)(CCO)CN(C(=O)N(C)C2CC2)C1 C=CC1(NC(N2CCCN(C(c3c(F)cccc3F)=O)CC2)=O)CCOCC1 N1(C(COCC(C)(C)C)=O)CCN(C(c2ncsc2C2CC2)=O)CC(O)C1 N1(C(C(CC)NC(N)=O)=O)CC2CCC(C1)N(C(=O)Cc1csnc1C)C2 c1(C(=O)NCC2C(C)CCN(C(c3cnn(C)c3Cl)=O)C2)coc(S(N)(=O)=O)c1 c1(C(=O)NCCOCCCNC(=O)C(F)=C2CCC2)ccc2c(c1)CNC(=O)N2 N1(C(COCc2cn(C)nc2)=O)CCC(NC(=O)CS(=O)(=O)N(C)C)C(F)C1 C=CC(CCC)CC(=O)NC1COC2(CNC(c3csc(Cl)c3)=O)CC1C2 Cc1sccc1CC(=O)N(C)CCOCCCN(C(=O)CC1CCOC1C)C c1(NC(C2CC(CCNC(=O)COCc3cccnc3)C2)=O)nc(C2CC2)cs1 Cc1ccc(F)c(C(=O)NCC(C)CNC(=O)Cc2n[nH]c(=N)s2)c1S(N)(=O)=O C(=O)(C#CC(C)(C)C)N1CC(n2cc(CNC(c3ccc(CC)[nH]3)=O)nn2)C1 N1(C(c2n(CC)c3c(c2)cccc3)=O)CCC2(CCN(C(=O)C3=NOCC3)C2)C1 N1(C(c2c(CCC)n(C)nc2)=O)CCCN(C(=O)C(C)C2CC2)C(CO)C1 C=CCN=c1[nH]cc(C(N2CCC(C3CCCN3C(=O)C(C)COC)C2)=O)s1 C1(NCC(C)(O)NC(COCCOCCOC)=O)CCN(C(=O)CC2CC2)C1 C1(C(=O)NC2C(CC)N(C(=O)Cc3ccc(Cl)cc3C)CC2)CC2(CCCC2)C1 c1(CCC(=O)NCCCC(CCC)NC(=O)CC(C)(C)O)cccc([N+](=O)[O-])c1 c1(C(N2C(CNC(CC(C)C(F)F)=O)CCCC2)=O)n[nH]c2c1COCC2 CC1CCN(C(=O)C=CI)C1CNC(c1cnsn1)=O C(=O)(CC(F)(F)C(C)(F)F)NCCOCCOCCNC(C=C(C)I)=O C12CCN(CC1O)Cc1ccc(cc1)NC2=O.c1(C(=O)OC)nc[nH]c1NC=O CC(F)(F)CCC(=O)NC1CC1CNC(c1ccc(Cl)cc1)=O N(C(=NCCc1nc2ccc(NC(C)=O)cc2o1)N1CCC(OC)C1)C(CC)C C(C(C)C(=O)NCC1CCOC1C(=O)NC(C)C(F)(F)F)OCC Cc1oc(C)c(C(=O)NC2CN(C(=O)CC(C)C3CC3)CC2C)c1C Cn1cnc2c(C(=O)NCC3CC(F)CN3C(=O)CC3CC(=O)C3)n[nH]c2c1=O c1(OC)cc(C(=O)OC)ncc1F.N12CC(CC1=O)CNCCC2 C1(CC)CCC(C(N2CCCC(C(=O)NC(C)C(C)(C)CN(C)C)C2)=O)CC1 CCCCCCC(=O)NCC(C)(CC)C(=O)NCc1ccccc1C c1(CC(=O)NCC(CNC(C(CC)(F)F)=O)C)c[nH]c2cccnc12 c1(NC(c2n3cc(C)sc3nc2)=O)nc2c(s1)C(C)(C)CC(C)(C)C2 C(N=c1nc2sccc2c(NCC(=O)NC2CC2)[nH]1)c1occ(C)c1 c1(C(=O)NC(CC)CN(C)C(c2cocc2C)=O)n[nH]c2c1CC(C(C)C)CC2 c1(OC)ccc2c(c1)C(C(=O)NCCCN(C)C(c1cnc(C#N)s1)=O)CCC2 C1(C)(CC)CCN(C(=NCCC(=O)NC)NCC2(O)CCCCC2)CC1 c1(C(=O)NC(C(C)NC(c2nn(CC)c(C)c2)=O)C)cnc2c(Br)cccn12 c1(OC)cccc(C(F)(F)C(=O)NC2CC(C)N(C(c3ncncc3F)=O)C2)c1 c1(C(=O)NC2CCCCC2)ccccc1NC(=O)CN1CCNCC1 C1(CNC(C2(CC=C)CCOCC2)=O)(OC)CCN(C(=O)COCC)CC1 O=C(CC1CC(F)CN(C(=O)CC2CSCCO2)C1)Nn1cncn1 C1(C(=O)NCCCN(C(=O)CC2OCCCC2(C)C)CC)CCC(=O)N(C)C1 c1(C(C)C(=O)NC2CN(C(c3ncncc3F)=O)C2)ccc([N+](=O)[O-])cc1F C12(NC(c3c(CC)occ3)=O)CCC1CN(C(=O)CCC(F)(F)F)C2 C12(C(=O)NCC3(CO)CCN(C(=O)COc4ccccc4)C3)CCCN(CC1)C2 c12ccc(cc1)C1(CCC1)N2S(C)(=O)=O.N1(C(C)C)CCCOCC1 Cc1ccc(CN2CC=CC(Cn3cc(-c4cncc(C)n4)nn3)C2)c(F)c1 c1(C(C)(C)C)ccc2cc3ccc(-c4ncc(CCOC=O)[nH]4)cc3nc2c1 C(=O)(C(O)C(F)(F)F)NCCC1CC(OC)CN1C(c1ccc(C#N)s1)=O c1(CN(C(=O)CCNC(N)=O)CCNC(C(C)NC(N)=O)=O)ccccc1Cl C1(C(N2C(CNC(Cn3nnc(C)n3)=O)COCC2)=O)CCCCC(=O)C1 C1(C)(C(=O)NC(c2cccc(C)c2)CNC(c2cc[nH]n2)=O)CCCCC1(F)F C1(CNC(C2(C(=O)OCC)CCC2)=O)COC(CNC(=O)C(C)OC)C1 N1(C(C2(C(N)=O)CCC2)=O)CCN(C(=O)CN2CCCCC2)C(CCO)C1 C(=O)(CCC(=O)N1CCCC(C(C)N)C1)N(CCN(C)C)CC.CCC c1(CNC(CC2(C#N)CC2)=O)ccc(CNC(C2(F)CC=CCC2)=O)c(F)c1 N1(C(C)C)CCOC(C(=O)N(C(CNC(=O)CCc2ccsc2)C2CC2)C)C1 C1(CC(=O)NCCCC2CC(C)C2)CCN(C(C2(Cl)CC2(F)F)=O)C1 Cc1cn(CCO)cc1NC(COC1(C)CN(C(=O)CC2CC3CCC2C3)C1)=O C1(NC(c2c(CCC)nco2)=O)CC(C2CCN(C(C3CCC(C)O3)=O)CC2)C1 CC(Cc1ccnn1C)C(=O)NCC(O)CCNC(C1COC(=O)O1)=O c1(C(=O)NCC2C(C)CCN(C(COC(C)C)=O)C2)ncnc2ccsc12 C#CCC(C)C(=O)N1CC(c2cc(O)n[nH]2)C1.C1C(C)CCN1C(=O)OC(C)(C)C c1(C(=O)NC(C)C(C)NC(=O)CC(C)(C)F)coc2c(F)cc(Cl)cc12 CC(C)S(=O)(=O)CCNC(c1ccncc1)c1nnnn1CCCC1CC1 CC1CN(C(c2n[nH]cc2CNC(c2ccccc2O)=O)=O)CC(=O)N1 N1(C(C2(C)CC(C)C2)=O)CCOCC(NC(=O)Cc2cncc(O)c2)C1 N1(CC(C)C)CCC(C(=O)NCCCCNC(=O)C(C)C2CC2)C1 c1nc(C(C)C)nn1-c1ccc(C2CC2)cc1.CC(C)CCCn1cc(CC)nn1 CC(C)S(=O)(=O)C(C)C(=O)N1CCC1CNC(c1ccccc1C1CCCC1)=O c1(CCNC(=O)Nn2ncc(NCCN(CC)CC)c2)c[nH]c2c(Br)cccc12 N1(C(C(C)SC(C)C)=O)CC(C)C1C(=O)NCC1CCCSC1 N1(C(CSCc2nc(C)sc2)=O)CC2CCC1CN2C(C1CCCC(=O)O1)=O Cc1[nH]nc2c1CC(C(=O)NC1CCCCCN(Cc3ccncc3)C1)CC2 c1(SCC(N2C(CNC(C3(C)C(C)(C)C3)=O)C=CC2)=O)cc(Cl)cc(Cl)c1 C1(NC(CCC(=O)OCC)=O)CCC2CCN(C(C3CCC(C)(C)CC3)=O)C1C2 C(=O)(CC(c1ccccc1)SCC(F)(F)F)NC(C)(C)CF C1(NC(C2N(C(CC(=O)NCC)=O)CSC2)=O)CCN(C)CC1(C)C c1(C(c2n(CCSC)nnn2)NCCCS(C)=O)nc(C)n(C)n1 C(CCC(O)C(=O)NCC(C)O)NC(C1(COC)CC(=O)C1)=O CC1C(C)N(C(c2cnn(C3CCC3)c2)=O)CCN1C(=O)Cc1cnco1 C1(OC)CN(C(=O)CCCC2CC2)CC1NC(=O)C(C)(C1CC1)OC c1(C(C(=O)N(C(CC)CNC(=O)Cc2nncn2C)C)O)cn(C)nc1C O=C1CN(C(C2CC3CC3N2C(c2ccc(N3CCCC3)cc2)=O)=O)CCN1 Cc1ccc(CN2CCC(NC(=O)COc3ccccc3C)C2)c(Br)c1.CCO Cc1c(N)c(C(N2CCC(NC(c3nccc(Cl)c3Cl)=O)C2)=O)nn1C c1(C(=O)NCc2ccc(C(N(CC(C)SC)C)=O)s2)ccc(C)cc1C C(=O)(C(F)C(C)(C)O)NC(C1CCN(C(c2cc(C(=O)OC)sn2)=O)CC1)C N1(C(c2c(CC)cco2)=O)CCN(C(=O)C(c2cc(C)oc2C)C)CC1CO C1(OCC)CC(C)(C(N2CC(=CCNC(=O)C(C)OCC3CC3)C2)=O)C1 CN1CCOc2c(C(=O)NC3CCC3NC(c3cncc(C#N)c3)=O)cccc21 c1(C(N2CC(CCC=C)(C(=O)N(CCCO)CC)C2)=O)c[n+]([O-])c(C)cn1 CC(CC1CCCCC1)C(=O)N1CCC(CNC(=O)CC2CC(C)(C)C2)C1 c1(OC)ccnc(F)c1C(=O)NC(C)CCCNC(C1CC(C)=NO1)=O C(CO)(CCCCNC(c1n[nH]c(C2CC2)c1Cl)=O)NC(C1C(C)(C)CCC1)=O n1(CC)ncnc1C(C)NC(CC(C)C)C1CCCCC1 CC(C)(C)C(C)(C)C(=O)N1CCC(CNC(=O)C(O)Cc2ccccc2)CC1 C(=O)(C1OC(=O)c2ccccc21)N1C(CNC(CCC2COC(C)(C)O2)=O)CC1 c1(C(=O)NCC(CO)NC(Cc2c(C)ccs2)=O)ccc(NC(C)=O)cc1F N1(C(=O)OC)CCCN(Cc2c(Cl)cccc2I)CC1 c1(C(=O)NC2C(NC(CN(CC)CC)=O)COCC2)ccc(F)c2c1CCC2 c1(CN2CC3C(C(=O)OC)(CCC3)C2)cc2c(C)cc(C)nc2s1 N1(C(CCC(=O)OCC)=O)CCCC(C2CCCN(C(C3CCC(C)C3)=O)C2)C1 C(=O)(C(CCCC)N(CC)CCOC)N(CC(F)(F)COC)CCC CC1CCC(Cl)=C(C(=O)NCC2C(C)CCCN2C(=O)C=CCn2cncn2)C1 n1(C(C)C)ccc(C(N2CCC(NC(=O)C3=COCCO3)C(C)C2)=O)cc1=O c1(C(=O)NCC2(F)CC(CC(=O)OC)C2)cc(C)n(C(C)C)n1 c1(C(N(C(CC)CNC(c2ccc(C(C)C)o2)=O)C)=O)noc(CC)c1C CC1(C)CCC(C(=O)NC2CN(C(C3CCCSC3)=O)CC2F)C1 N1(C(c2c(C)coc2)=O)CCC(N(C)C(C2Cc3ccccc3O2)=O)C2(CC2)C1 C1(C(=O)NCC(C(C)C)NC(C(CC)SC)=O)CC2CCC1O2 N1(C(CCC)=O)CC2CC(C(=O)NC)CC2C1.c12ccc([nH]1)NC(=O)CC2 C1(C(=O)NC(C2(O)CN(C(c3c[nH]cc3C3CC3)=O)C2)C)CC2(C1)CC(O)C2 c1(C(C)N(c2cn(CC(F)(F)F)nn2)C(=O)C(C)(C)F)cc(F)cc(F)c1 c1(C(=O)NC(C(C)C)CNC(C2(CF)CCOCC2)=O)cc2ncccc2[nH]1 CCC(C(O)C(F)(F)F)NC(c1cc(-c2cnn(C)c2)cc(N)c1)=O c1(CN(C(=O)CCCF)C)ccc(CNC(=O)CCc2ccc(O)nn2)cc1 c1(OC)cc2c(cc1OC)C(NC(c1ncccc1Cl)C)CC2 N1(C(C)CC2CCCCC2)CC2COCC2(C(N2CCC3(C2)CC3(F)F)=O)C1 C12(NC(Cc3ncc(C)s3)=O)CCCCCC1N(C(c1cnc[nH]1)=O)CC2 c1(OC)c(NC(C2CC23CN(C(=O)C(C)NC(C)C)C3)=O)cnc2ccccc12 C1(C(N2CC(n3cc(CCCC(F)(F)F)nn3)C2)=O)CCc2nncn2CC1 C1(C(C)C(=O)N(C)CCC2CCCO2)CCN(C(c2ccc(CO)cc2)=O)CC1 N1(C(C(C)OCC#C)=O)CCCC2C1CCN2C(c1cc([N+](=O)[O-])ccc1Cl)=O C1(C2CCC2)(C(=O)NCC2CC(F)(F)CN2c2cnc(F)cn2)CC1(F)F Cc1nc(C)c(C(=O)NCCC(O)CNC(c2c[nH]cc2C(F)(F)F)=O)s1 C1(CNC(C(C)CC2CCCCC2)=O)CC(F)CN1C(c1ccc(Br)o1)=O N1(C(c2ccc(OC)s2)=O)CCC2CN(Cc3cccc(F)c3Br)CC12 c1(C(N2CCCN(C(Cn3c(C)ccn3)=O)CC2C)=O)c[nH]c2c(F)cccc12 c1(C(N2CC(CC(=O)Nc3c(C)ccnc3Br)C2)=O)c(Cl)cnc(Cl)c1Cl C1(CNC(CN(C(=O)OC)C)=O)CCN(C(C2C=CC=CC=C2)=O)C1(C)C N1(C(c2ccc(CC(C)C)cc2)=O)CC2(C1)SCCC2NC(C1CC1F)=O c1(C(=O)NC(CN(C(C(C)NC(CC)=O)=O)CC)C)ccc2nnc(S)n2c1 C1(NC(CC2CC(=C)C2)=O)CC2CCC1N2C(c1n[nH]c(C(C)(C)C)n1)=O CCCC(C)(C)C(=O)NCC(C1CCCC1)NC(C1(Br)CC12CCC2)=O c1(C(C(=O)N(CCNC(C(C=CC)O)=O)C)(C)OC)ccc(OC)cc1 CC1CN(C(=O)C2=CCC2)CCCN1C(=O)CC(C)(C)Cc1ccc(Cl)cc1 c1(NC(c2nc(NC(c3ccc(OC)nc3)=O)sc2)=O)ccc([N+](=O)[O-])c(F)c1 N1(C(CCCCOCC)=O)CCC(NC(c2cc(C#N)oc2C)=O)C2(CCC2)C1 c1(C(N2CCOC3CCN(C(C(C)SC)=O)CC32)=O)cnc2ccc(F)cc2c1 CCCC(C(=O)NC1CC(F)(CNC(C2(C)CCOC2)=O)C1)C(C)C c1(C(=O)NCC2C(NC(C=C(CC)C)=O)CCCC2)ccc2cc[nH]c2n1 C1(CNC(CC2CC(=C)C2)=O)(OC)CCN(C(=O)C(C)(C)C2CCOC2)CC1 C1(F)(CNC(C(C=C)OC)=O)CCCN(C(=O)C(O)CC2CCCC2)C1 c1(OC)ccc(CN2CC3CN(C(c4cccc(I)c4C)=O)CC3C2)c(F)c1F C(N=c1nc2scnc2c(NCc2nncn2CCC2CC2)[nH]1)c1cc(CC)on1 C1(OC)CC(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCC2)N(C(C)=O)C1 O=C(N=c1ncn(C2CC2c2ccccc2)[nH]1)Nc1cc(F)cc(F)c1 C(CO)(CO)(C(=O)OC)NCC(CCCC)c1ccccc1C(F)(F)F C1(C(N2CCC(C(C)NC(C3CN(C)C3)=O)C2)=O)CCC(=O)N1C N1(CCC(CC)O)C(=O)NC(CCCc2ccccc2)C1=O N1(C(COCCCC)=O)CC(F)(F)CC1(C)CNC(C1CCC(CCO)CC1)=O C1(C(C)C)CCOC1C(=O)NCC1CN(C(=O)C(C)CC2CCC2)C1 c1(C(N2CCN(C(=O)C3=CSCS3)C(CO)C2)=O)cc2ccsc2s1 c1(C(=O)NCCCCN(C)C(C2(C)C=CCC2)=O)ccn(C)c1 c1(C(=O)NCC2N(C(C(c3n(C)cnc3)O)=O)CCC2)ccc(SC2CC2)nc1 Cn1c(NC(=O)NCC2(N3CCOCC3)CCCOC2)cnc1S C(N=c1[nH]c(C)ncc1C)C1CCC(NC(C(CCC)N(C)C)=O)C1 N1(C(CCC2C(C)(C)C2)=O)CCC(O)(CNC(=O)Cn2ccc(O)nc2=O)CC1 c1(C(=O)Nc2c(CC)nn(CC)c2)cc2cccc(C(F)(F)F)c2nc1O c1(C(=O)NC2C(C(N(CCCOC)C)=O)CCC2)ccc(C)nn1 C1(N(C)C(c2nsnc2O)=O)CCCC(NC(=O)C(c2ccc(F)cc2)(C)F)C1 c1(C(N)=O)ccnc(C(=O)NC2C3CN(C(C4CCCS4)=O)CC23)c1 Cc1ccc(C)c(C(=O)N(C)CCNC(=O)CCNC(c2ccncc2)=O)c1O CC1=C(C(=O)N2CC(CN(C(=O)C(O)C3CC3)C)C2)Cn2ncnc2N1C c1(OC)cccc2c1C(C(=O)NC1CCN(c3ccc(C)cn3)CC1)CC2=O C(CCCC(=O)NC1CC(F)(CNC(c2ccc(CC(N)=O)cc2)=O)C1)OC C1(C#N)(CNC(c2c(C)nc(CNC(C3CCCC(C)C3)=O)o2)=O)CC(C)(C)C1 N1(C(CC2CC(C)(C)C2)=O)CC(NC(C2(C)CCC(=O)N2)=O)C(n2ccnn2)C1 C12(NC(CC(=O)NCC)=O)CC(C)(C1)OC21CN(C(C2COCC(C)O2)=O)C1 C1(C(=O)NCC(C)N(C)C2CC2)CCC(C2CC2)N1C(=O)Cc1ccsc1 C1(O)(CCNC(=O)CC2CC3(CC3)C2)CCN(C(c2ccnc(C3CC3)n2)=O)C1 C(=O)(C(CC(N)=O)NC(=O)CCCCN(C)C)NC(C=C)(C)C CCC(CC(=O)N1CCCC1CCNC(=O)C(c1ccc(OC)cc1)C)OC C1(NC(c2c(C)occ2)=O)CCCCN(C(c2cn(C)nc2C(F)(F)F)=O)C1 C1(C(=O)OC)CCCN(C(=O)C(C)(C2CC2)N(C(=O)CCN2CCCC2=O)C)C1 N1(C(Cc2c(C)n[nH]c2)=O)CCCN(C(=O)C(C)(F)F)C(C)C1 C1(C(=O)NC(CC#C)CC(F)F)CN(C(=O)C(CC2CC2)OC)CC(C)(C)C1 Cc1cncc(C(N2CC(CNC(=O)CCc3nc(C4CC4)no3)C3CC23)=O)c1 c1(CCC(=O)N(C(=O)C2=NOCC2)C)c(C(F)(F)F)oc2ccccc12 CCCCC(CNC(=O)C=Cc1ccco1)NC(=O)CCCCF C1(C2CCC2)(C(=O)NCc2c(CN(C)C(c3ccc(Cl)o3)=O)cccc2)CC1 O=C(CN1C(=O)Cc2cc(Cl)ccc21)N1CC(n2cc(CO)nn2)C1 CCCC(C)C(C)N=c1nc2c(cnn2C(C)C)c(NCCC(C)(C)C)[nH]1 CN1CC2CC1CN(C(C1(NC(c3cc4cccn4cn3)=O)CCCCC1)=O)C2 C12(NC(c3ccnc(C)c3C)=O)CCCCCC1N(C(=O)COC(F)(F)F)CC2 C1(N=[N+]=[N-])(C(=O)NC(c2ccco2)C)CCN(C(c2ccccc2)=O)C1 C(=O)(C1CCCc2nncn21)N1CCC(CCNC(C(C)c2cccs2)=O)CC1 c1(C(=O)NCC2CN(C(c3c(C)nc(O)[nH]3)=O)C2)cc2cnc(C)nc2nc1O Cc1c[nH]nc1COCCN(C(=O)C(c1ccnn1C)O)C.N1(C)CC1 c1(C(=O)NCCC2(O)CCN(C(C3C(C)C3)=O)C2)ccc2c(c1)NCCC2 Cc1cc(C(=O)NCC=C2CCN(C(C3CC3C)CC=O)CC2)cc(N)c1 n1(CCC(N2C(CC)CN(C(=O)Cc3cccs3)CC2)=O)c(C)cc(=O)cc1C C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(c2cncc(C)c2)=O)C(C)CC1 C1(C(=O)NC2CC(OCC(=O)NCc3cn(CC)nc3)C2)CCN(C)C1C N(C(=NCCCCl)NCCOc1cccc(F)c1O)CCC1C(C)(C)CCO1 N1(C(N(CCCC)C)=O)CCCC(C(=O)NCC(C)(O)C(F)F)CC1 N1(C(CCC=C)=O)CCOC2(CCN(C(=O)C(C)(F)C(=O)OC)C2)C1 N1(C(C(F)=CC)=O)CC2(CCN2C(=O)CCCC2CCCCC2)C1 c1(CN(C(=O)C(C2CC2)NC(C2CCCSC2)=O)CC)cncn1C C(=O)(NN1CCCC1NC(=O)NCc1c(OC)cccc1)C1CC(C(C)(C)C)=NO1.N C1(NC(=O)NC(c2ccc(CCC)cc2)C(C)C)(CSC)COC(C)(C)OC1 c1(N2CCC(N(CCC)C(C3CC3(C)C)=O)CC2)snc(Cl)c1C#N C(=O)(CCCCC(C)CC)NC1CCC(C(N(OCC)CC)=O)C1 C1(NCC(C)(C)OC)CC(Oc2nnnn2C2CC2)C12CCC2 N1(Cc2cn(C(C)(C)CCCCn3ccnn3)nn2)CC(=O)CCC1=O c1(C(=O)NCC2CCC2)ccc(OC)cn1.C1(CCNC=O)(CC)CCCC1 C12(CNC(C3N(CC)CC3)=O)CC1CN(C(=O)Cc1c(Cl)cnn1C)C2 CC(N=c1nc2scnc2c(N2CC(CO)C2)[nH]1)c1nc(=N)[nH][nH]1 N1(C(C=CC(C)(C)NC(=O)C=CCO)=O)CCC2CCC(C2)C1 C(=O)(CCC(C)OC)NC(CC)CNC(C1CC1COC)=O Cc1cc(=NCc2cncs2)[nH]c(=NC(C)CN2CCOC2=O)[nH]1 c1(OCC(C)NC(COCC(=O)OC)C)ccccc1.C(C)(C)O N(C1COc2cc(Br)ccc21)c1nccc(=NC(C)c2c(CCC)nns2)[nH]1 C1(CN(CCCC)CCCC(O)C(F)(F)F)(CNCc2ccccc2)CC(F)(F)C1 N1(C(CN(C(=O)CC2CCCC(C)C2)CCOC)=O)CCCC(C)(C)CC1 N1(C(c2c(OC)nn(C)c2)=O)CCC(O)(C(=O)N(C)CCn2cccn2)CC1 c1(C(N2CCCC(Oc3cccc(CO)c3)C2)C#N)c(Br)cc(Br)cc1Br C1(NC(C(C)SC)=O)CN(C(c2c(O)cccc2O)=O)CCC1C C(=O)(C(F)(F)C(O)C1CC1)NCC1CN(C(=O)C=CSc2ccccc2)CC1O n1(C(C)C)ncc2c(NCc3cscn3)[nH]c(=NC3CCCC3C(C)C)nc12 C(c1cnc(C)nc1O)=CC(N1C(CO)CC(NC(COC(CC)C)=O)C1)=O CN1CC(C)(C)CC1C(=O)NCC12CC(CO1)N(C(C1CC(C3CC3)=NO1)=O)C2 N1(C(COCCC)=O)CC2CC2(NC(c2ccccc2C2CCCC2)=O)C1 N1(C(C(N2CC(CC(N3CC(CC(=O)OC)C3)=O)C2)=O)C)CCCCC1=O C12(C(=O)NC3CC(NC(c4cccn(O)c4=O)=O)C3)CCCC1OCC2 N1(C(C(C=CC)O)=O)CCN(CCNC(C2CN(C(C)=O)C2)=O)CC1 O=C(C1=NOCC1)NCc1cc(C(N2CCOCC2CO)=O)co1 C1(NC(c2cc(C(C)=O)on2)=O)CC(C(=O)Nc2ccsc2)C1(C)C c1(C(N2CCC(C)C2CNC(c2cnc(O)n2C)=O)=O)ccn(CCO)c(=O)c1 C1(CNC(C(C)OCC=C)=O)CCN(C(=O)CSc2cccc[n+]2[O-])C(C)C1 N1(C(C(C)CCN(C)C)=O)CCC(C2(NC(=O)CC(C)SC(F)(F)F)CC2)C1 c1(CNC(N2CC(c3nc(C(=O)OC)c(C)s3)C2)=O)ccc2nc(C)oc2c1 c1(C(=O)NC2CC(CNC(C3ON=C(C)C3)=O)C2)[nH]cc2c1CCC2 c1(C(=O)NC2CC(C(C)NC(C(CC)O)=O)C2)cc(O)ccc1Cl C(C)(CNC(c1cnc(S)n1C)=O)(CC(C)C)NC(COCCCC)=O C(=O)(C1=C(C#N)CCC1)N(CCCNC(c1cc(C(F)F)cs1)=O)C(C)C c1(C(=O)NCCC2CCC(NC(=O)Cc3ccco3)C2)ccnc2ccnn12 C#CC1(O)CC(C(=O)NCCC2(NC(C3(O)CC3)=O)CC2)C1 C1(C(N(CC(=O)N(C)CCC2CCCN2C)C(C)C)=O)CC2(C1)CC21CC1 C12(NC(=O)Nc3c(N)c(Cl)ccc3)CCC(Cc3cnn(CCl)c3)(CC1)OC2 N1(C(CC(C(=C)C)OOC)=O)CC2CCCC(N=c3ccnc(OC)[nH]3)C2C1 c1(CC(N2CC(CN(C)C(C3C4COCC34)=O)C2)=O)cnn(C)c1 C(=O)(C1=C(Cl)CCOC1)N1CCN(c2nnc(C(C)C)o2)C(C(C)C)C1 N1(C(C(C)(C)CCCO)=O)CCCC(C2CCCN(CCF)C2)C1 C1(NCc2nnc(C)o2)CC(NC(c2cc(Br)c[nH]2)=O)C12CCC2 C=CCC(C)(C)CC(=O)NC12CC(C(=O)N(CC(C)C(C)(C)C)C)(C1)C2 C(=O)(CCCC(C)(F)F)NC1CN(C(c2cnn(CCC)c2C)=O)CC1C C(=O)(C1=C(C)CCOC1)N1CCN(C(CC2CC(OC)C2)=O)CC1.C(COC)N C1(NC(=O)CC2(C(F)F)CC2)CCCN(C(c2nnc(O)cc2O)=O)CC1 C1(C(=O)Nc2cc(OC)cc(O)c2)CCN(C(=O)C(C)(C)C(N)=O)CC1(C)C C1(NC(CCSC)=O)CCC(C(=O)NCCC(C)(C)SC)C1 c1(C(=O)NCC(CC)NC(=O)CNC(c2cccs2)=O)coc2c(C)cccc12 C1(C(N2CCC(COC)C2)=O)CCC(O)CN1C(=O)CN(C1CCC1)C C(=O)(C1=CCCOCC1)NCC(C)N(C)C(C12CC(C1)C2)=O c1(-c2n(CC)c(N3CCCC3Cn3ccnn3)nn2)cn2ccc(C)cc2n1 N1(C(c2cc3occc3[nH]2)=O)CC(C2CCCN(C(C34CCC(C3)OC4)=O)C2)C1 C(=O)(C1=CCCC1C)NC(C(=O)NCC(CC)CO)Cn1cncn1 C1(NC(c2c(C)ccnn2)=O)CC12CCN(C(C1CCCC13CCC3)=O)C2 CC1(C)CN(CCn2cc(S(C)(=O)=O)cn2)Cc2ccc(Br)cc21 C(c1cncc(C)c1)=CC(N1CC(CC=C)(C(=O)NC(C)CC2CCOC2)C1)=O CC1=C(C(=O)NC2(C)CC(NC(c3[nH]nnc3C)=O)C2)CC1 C1(C)(NC(CCN(C(CCC)C)C)=O)CC(NC(=O)CCCc2ncc(C)o2)C1 CC1(CNC(c2ccc(OCC(F)F)nc2)=O)CCN(C(C2CCCS2)=O)C1.C S(=O)(=O)(c1ccc(C#N)cc1)N1CCC(NCc2cc(C(=O)OC)no2)CC1 N1(C(CCOCCC)=O)CCC(CNC(c2ccc(C)c(O)n2)=O)C(C)C1 C=C(C)CC(C(=O)NCCCCc1cn(CCCOC2CCC2)nn1)OC C1(CCC(=O)N(CCOC)CCNC(c2cn(C)nn2)=O)CCN(C)CC1 O=C1C2COCCN2C(=O)N1Cc1ccc2cnccc2c1 C1(NC(c2nccc(C)n2)=O)CCN(C(c2ccncc2Cl)=O)C12CCC2 CC(CCC(=O)NC1CCN(C(=O)C#CC2CC2)C1C)c1ccccc1 N1(C(CCCC(C)(C)C)=O)CC2CN(C(C3(C)CCCCO3)=O)CC(C1)O2 c1(CS(=O)(=O)N(CC(C)C#N)C)ccc(F)cc1F C12(C(N3CCC(O)(C(C)NC(=O)Cc4ccco4)CC3)=O)CCC(F)(CC1)CC2 N1(C(C(C=C)CC)=O)CCC(C=C)(C(N2CCC(CC)CC2)=O)C1 C1(NC(C(C)OCC)=O)CCSC12CN(C(c1ccsc1OCC)=O)C2 c1(C(N2CC3C(C(N4CCC(F)C4)=O)C3C2)=O)cc(Br)cc2cn[nH]c12 C1(C(CCCC)c2nnnn2C2COC2)=CCC(N=[N+]=[N-])C1.C(C(C)C)N N1(C(C2(C)CCN(C(C(CC)OCC)=O)C2)=O)CCCC(C)C1CO C(=O)(CC(F)(F)C(F)(F)F)N1CCC2(CC(NC(c3c(C)nn[nH]3)=O)C2)C1 c1(C(=O)NCCCN(C(c2c(SC)ccs2)=O)CCO)cccc(F)c1C1CC1 C1(CNC(CCN(CC)CC)=O)Cc2ccccc2O1.C(C)(C)O N1(C(CN(C(C)=O)C)=O)CCC(C2CCCCN2C(=O)CC2CC2(Cl)Cl)CC1 C(C(C)(C(=O)O)NC(=O)CC(=O)Nc1ccc(N)cc1)OCC c1(CN(C(c2c(CC)occ2)=O)CC2CCCC2)c(C)nn(-c2ccccc2)c1Cl C1(O)(CCNC(Cc2nc(C)sc2)=O)CCN(C(=O)Cc2ccncc2Cl)C1 Cc1nn(C)c(C(F)(F)F)c1C(=O)Nc1ccccc1CN1CCOCC1 Cn1ccc(C(=O)NCC(C)(C)CNC(=O)Cc2ccns2)c1C1CCC1 C(=O)(CC(O)CC(C)(C)C)NC12C(CN(C(c3c(COC)noc3)=O)C1)CC2 Cn1cnc2c(C(N3CCCC(C(F)(F)F)C3)C(N3CCOCC3)=O)cccc12 C(C(=O)NC(C)CNC(c1cc(C2CCOC2)[nH]n1)=O)(C(C)C)NC(COC)=O N1(C(CC2CC(CC)OCC2)=O)CCC(C2CC2)C1CNC(=O)CCNS(C)(=O)=O c1(C(=O)NC2CCC(N(C(=O)CN3CC=CC3)C)C2)ccc(Cl)cc1N c1(NC(C)=O)cc(C(=O)NCC(C)(C(C)C)NC(=O)C(C)C(F)(F)F)ccc1F C(=O)(C1CCCc2sc(C)nc21)N.CCCCCCCNC(=O)CCN(CC)CC C1(C(N(CCC(C)NC(c2cn(CCOC)nn2)=O)C)=O)CN2CCN1CC2 c1(C(=O)NCCN(C(CC2C(C)C2)=O)C2CC2)cc(-c2ccccc2)no1 N1(C(CC(=C)Br)=O)CCCCC1CCNC(=O)COC1CCCOC1 C1(CCNC(C(C)OCC(C)C)=O)CCN(C(c2nonc2N)=O)C1 CC(N=c1[nH]c2c(c(=NC(C)Cc3cn[nH]c3)[nH]1)SCC2)C1CSCCO1 N1(CC(C)(C)NC(C2C(C)(CC)C2)=O)CCN(C(c2ccccc2SC)=O)CC1 N1(C(CCC)=O)CC(F)CC1C(=O)OC(C)(C)C.C12(C)CC1CNC2=O.OCSC c1(OC)ccc(CC(=O)NCC(C)N(C)C(c2cc(Cl)n(C)n2)=O)c(Cl)c1 c1(NCC2C(C)C2C)ccc(S(=O)(=O)N2CC3C4C=CC(O4)C3C2)cc1F c1(C(N2CCC(C(=O)NCC(CCC)C#N)C2)=O)noc2c1CN(C(C)C)CC2 N1(C(c2scc(C)c2)=O)CCc2ccccc2C1CNC(c1ccccc1Cl)=O c1(OC)ccc(NC(C2C=CCN2Cc2ccc(-c3ccccc3)s2)=O)cc1C c1(C(C(=O)NC(CC)(C)C)N(C2CC(F)(F)C2)CCCO)ccc(Cl)c(Cl)c1Cl C12CCN(CC1(F)F)C(=O)NC2.c1(CNC(=O)CO)ccc(Cl)c(Cl)c1 c1(C(=O)NCc2cccc(SC)c2)cc2cc(-c3sc(C)nc3C)ccc2o1 C1(CNC(CC=CC=C)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)C12CC2 C1(COCC)CCN(C(C2(NC(c3c[nH]cc3C)=O)CCCC2C)=O)CC1 C(=O)(C(F)(F)C(F)(F)C(F)F)NC1CCC(N(C(C(c2ccn(C)c2)C)=O)C)C1 CCC(CC)C(=O)NC(C)C(C(C)C)NC(c1cnn(C(C)C)c1Br)=O c1(C(N2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)=O)cnn2cccc(Cl)c12 CC(CC(=O)N1CC(NC(c2cnn(C3CCCC3)c2)=O)C(C)(C)C1)C(F)(F)F CC1COCCN(C(C2CC(NC(=O)C(C)n3cccc3)C2)=O)C1 N1(C(CC23C(CN(C(CN(C)C(=O)C4CC4)=O)C2)CC3)=O)Cc2cccc(F)c2C1 c1(C(C(=O)NCCCC#C)N(CCC)CC)cnc(-c2ccco2)s1 C12(C(=O)NCCOC3CCN(C(CN(C)C)=O)CC3)CCOC1CCOC2 C=CC1CN(C(c2cn3c(n2)CCC3)=O)CC1NC(=O)CCCCc1cnn[nH]1 CCC(CCCO)NC(=O)CCCN(C(=O)CC=C(Cl)Cl)C c1(OC)cc(CN2CC3C(C2)N3S(=O)(=O)c2cccc(F)c2)cc([N+](=O)[O-])c1Cl c1(C(N2CCC(C3N(C(C(C=C)O)=O)CCC3)C2)=O)cccc(C)c1[N+](=O)[O-] CC1CCN(c2cc(C(N3CCC(F)(C(=O)NC4CCCS4)C3)=O)ccn2)CC1 n1(CCCOCC(CNC(=O)CCC2CCOC2)O)cc(CO)nn1 CN1CCC2CCN(C(C3CCN(C(c4cnn(C)c4)=O)C34CC4)=O)C2C1 N(C1CCc2cccnc21)C(C(C)CC(F)(F)F)=O C(=O)(C(C)(O)CCSC)NCC(C(=O)NC1(CC)CC1)CC1CC1 c1(OCC)cnc(Cl)[nH]c1=NCC1CCCN1C(c1cc(=O)c(OC)co1)=O C(=O)(C(F)CCC(C)C)NC.C(CC(=O)NC1CC(C(C)O)C1)SC C(=O)(CCC(=O)N1CCOC(CCNC(=O)C(C)COCC)C1)OCC N1(C(=O)OC)CCC(Cc2ccc(F)cc2)(Cc2cccc(O)c2)C1 c1(C(=O)NC2(C)CC(NC(c3c(C)csc3)=O)C2)cc(Br)n(C)c1 C1(C(=O)NCCCCCNC(C2(C)CCNC2=O)=O)Cc2n[nH]cc2C(=O)N1 C=CC(C)(C)CC(=O)N1CCCCC1C(=O)NC(C)C(O)C(F)F C1(CCNC(C(C)CN(C)C)=O)CCCN(C(c2nc(Cl)c(Cl)s2)=O)CC1 N1(C(c2cnco2)=O)CCOCC1C(=O)NCC1(CC(=O)OC(C)(C)C)CC1(F)F N1(C(CNC(CCC)=O)=O)CC(NC(c2ccc(CC)o2)=O)C2(CCC2)C1 C1(NC(=O)CCc2ccccc2F)COC2(CNC(=O)COC(F)F)CC1C2 c1(OC)ccc2cc(C(=O)NCC(C)CN(C)C(C3CCCO3)=O)ncc2c1 Nc1ncccc1NC(=O)Cc1csc(NC(=O)NCCc2ccc(O)nc2)n1 c1(C(N2CC(NC(CCOCCC)=O)CC2(C)CC)=O)cc2ccccc2nn1 C1(C(=O)NCCOCCCNC(=O)CCNc2ccsc2)C(F)(F)C12CC2 c1(C(=O)NCCCn2cc(CC(O)C3CC3)nn2)cccc[n+]1[O-] N1(C(CC(C)(C)C#N)=O)CCC(C2CC2)C1C(=O)NCc1cc(C2CC2)no1 CN1CCN(C(c2cc(F)cnc2O)=O)C(C(=O)NCC2(C)NC(=O)NC2=O)C1 N1(C(C2ON=C(C)C2C)=O)CCCC2(CCN(c3ccnc4ncnn34)C2)C1 c1(NC(N)=O)ccc(CC(=O)N2CC(C3CN(Cc4cnc(O)[nH]4)CCO3)C2)cc1 CCC(C(=O)NC(C)C=CC(=O)NCC(C)(O)C1CC1)N(C)C CC(C)(C(=O)NCC1(F)CN(C(=O)CCc2ccoc2)C1)C1CCCC1 C(N=c1[nH]c(=NCCCc2c[nH]nc2C)[nH]c2cccnc12)C1(CC)CC1 C1(NC(C(C)n2ccnn2)=O)CCN(C(C2(Br)CC2)=O)CC1F Cc1ccc(F)c(C(=O)NCCC(O)C(=O)NCC2CC(N(C)C)C2)n1 Cc1nc(O)ccc1C(=O)NCC(C)CNC(c1ccnc(-n2cccc2)c1)=O Cc1c(C(N2CC(F)CC2CNC(=O)C=CC(C)C)=O)nn2c1OCCC2 c1(CCCNC(N(C)CC2CC2(C)C)=O)ccnc(O)c1 C1(F)(CNC(C2CCCCC23CC3)=O)CCCN(C(=O)CSc2nncs2)C1 N1(C(=O)OC)CC2C=CC1C(C(=O)NCCN(C(c1cc(C)cnn1)=O)CC)C2 C(C(F)(F)CC(O)CO)N(C(c1cc(C)ns1)C(=O)N)C.C(C)(C)(C)O c1(C(=O)NC(CC)CNC(C2CCC(C)O2)=O)cc(OC)c(C)c([N+](=O)[O-])c1 CC(CC(=O)NCC1COC(CNC(=O)Cc2csc(=N)[nH]2)C1)N1CCCC1=O N1(C(c2[nH]n(C)c(=O)n2)=O)CCN(C(=O)CC2CSCCS2)CC1CCO Nc1cccc(C(=O)NC2CCCN(C(C3CC34CCOC4)=O)C2)c1N N1(C(C(CC)C)=O)CC2(CCCC2NC(=O)COc2cc(Cl)ccc2C)C1 N1(C(CC(C)=C(C)C)=O)CCOC2(CCN(C(c3ccc(Cl)nc3O)=O)C2)C1 C1(CCNC(Cc2nc(CC)sc2)=O)CCN(C(c2csc(C)c2)=O)CC1 c1(C(C(=O)NCC=C)N(C)CC2(C)CCCCC2)cc(Br)cc2cccnc12 N1(C(c2cc(C)on2)=O)CCC(NC(=O)Cc2ccc(O)cn2)C(C)(C)C1 c1(C(N(CCNC(CCCOCCOC)=O)C2CC2)=O)ncccc1SC.C1CO1 C(CC(C(=O)N1CCC(C(=O)NCC)C1)NC(C12CC(F)(C1)C2)=O)=CC C12(C(C(=O)C=CCN3CCCC3)=O)CCCN(c3nnc(C(F)(F)F)s3)CC1C2 Cc1cc(C)cc(C=CC(=O)NC2(CNC(c3cccnc3Cl)=O)CCC2)c1 C1(CNC(=O)CC2CCC2)CC2CC1CN2C(=O)Cc1ccnc(O)c1 n1(CCC)ncc(C(N2CCC(N(C(=O)C3=C(Cl)CC3)CC3CC3)CC2)=O)c1Cl C(=O)(C1=COCC1)NC1CN(C(C(C)C2(c3ccccc3)CCC2)=O)C1 c1(C(=O)NCCn2cc(CC(CC)(C)O)nn2)cc(C#N)ccc1Cl c1(C(=O)NCCN(C(C(CC(=C)C)C)=O)CC(C)O)cc2ccnc(Cl)c2s1 CCCCCCCCCC(=O)NCC1CC(NC(=O)CC2CCCOC2)C1 N1(C(c2c(C)ccs2)=O)C2CCC1C(C)C(NC(=O)Cn1cnc(C(N)=O)n1)C2 c1(OC)cccc(C(O)C(N2CC3CC3(NC(=O)CCn3cncn3)C2)=O)c1 C=C(Cl)C(C)(C)C(=O)NC1CCC(CNC(=O)COc2cc(C)ccc2F)C1 Cc1ccc(Cl)c(C(=O)NC2CC(F)CN(C(=O)C=Cc3ccc(Cl)nc3)C2)c1 c1(-c2c(OC)ncc(C(=O)NCC3CCO3)c2)ccc(O)c(C#N)c1 C1(C(=O)NC2(C(=O)OC(C)(C)C)CC(F)C2)(NC(C2CCCO2)=O)CCCOC1 c1(NC(CCCC(CCNC)C2(S(=O)(=O)CO)CCOCC2)=O)nc2ccsc2c(=NCC(N)=O)[nH]1 C1(NC(C=CC=CCC)=O)CC(CNC(c2ncccc2Cl)=O)C1(C)C C#CC1(C(N2CCOCC(C(=O)NCC3(C)CNC(=O)O3)C2)=O)CCCCC1 C(=O)(C1Cc2c(Cl)cccc21)NCC1OCCCN(C(CC(C(C)C)C)=O)C1 C#CCC(CC#C)C(=O)N1CC(N(C(=O)CSc2ccc(C)cc2)C)C(C)(C)C1 c1(CSC)cc(C(=O)NC(CNC(=O)Cc2cn[nH]c2)CO)ccc1F C1(NC(=O)Nc2cccc(-n3cnnn3)c2)CCCN(CC2CCCCCC2)C1 CC(C)C(CNC(c1cc(C#N)n(C)n1)=O)C(=O)NC1CN(C)NC1=O C(=O)(CC(C1CC1)NC(=O)C(CC1CC1)NC(=O)C=CC(C)(C)C)NC N1(C(CCC=C)=O)CCC2(CC(NC(=O)CCc3cnc4n3CCCC4)CO2)C1 c1(CCC(=O)NCC)cc(C)on1.C1(=O)CCCONC(=O)CC2CCCN12 N1(C(c2nc(CC)oc2)=O)C2CCC1CC(N(C)C(C1CCC3(CCC3)O1)=O)C2 Cc1cc(C(N2CCN(Cc3c(Cl)ccnc3Br)CC2)=O)ccc1F C1(C)(C(=O)NC2CCC(NC(C3(COC)COC3)=O)CC2)CCN(C)C1=O C#CC1CCCN(C(=O)C(C)(C)CNC(c2cnn(C3CC3)c2)=O)C1 N1(C(N2CCN(C(C3CCS(=O)CC3)=O)CC2)=O)CCC(Cc2ccccc2)CC1 N1(C(c2cn(C)c(=O)cn2)=O)CC2CCC(CNC(C3(C(N)=O)CC3)=O)C2C1 c1(C(C)N(CC(=O)O)C(c2cn(CCCF)nn2)=O)ccc(Br)cc1 C1(CC)COC(C)CN1C(=O)CN(C)C(c1n[nH]cc1C)=O c1(C(OCCCNC(c2nnnn2C(C)(C)C)(C)C2CC2)CC)ncc(Cl)cc1Cl C(CCCCCNC(=O)CC1CCCN1C(=O)C(C)CC=C)SC C1(NC(CCC=C(C)C)=O)CCCN(C(c2cccn2-c2ccc(F)nc2)=O)C1 c1(-n2cc(CN(C3CC(NC(CC(CC)C)=O)C3)C)nn2)ccc2c(c1)CCC2 c1(CC(C)C(N2CCCCC2CNC(=O)CC2CSC2)=O)ccccc1Cl N1(C(C=COCC)=O)CCN(CCN(C(=O)CSCc2ccc(F)cc2)C)CC1 CC1COc2c(C(N3CC4CCC(C3)N4C(=O)C(C)CF)=O)cccc21 C1(c2ccc(CC)cc2)CN(C(=O)CN2CCC2C)CCN1C(c1cn[nH]c1)=O C#Cc1ccc(C(N2C3CCC(C3)C2C(=O)N(CC(C(C)C)OC)C)=O)cc1C N1(C(c2cc(CC(C)C)on2)=O)CCCC(C(C)NC(c2cccnn2)=O)C1 CC1CCN(C(=O)CCc2cnn(C)c2)CC1CNC(c1ccc(Cl)c(F)c1)=O CN1CCCC(CC(=O)NC2(CCCC(=O)N3CC(CS(C)=O)C3)CCC2)C1 C1(NC(C(C)O)=O)C=CCN(C(c2cn(C3CCCC3)nn2)=O)C1 CC(C(=O)NCC1(O)CCN(C(c2ncoc2C(F)(F)F)=O)C1)C(C)(F)F C(C(=O)NCC(C)(C)CC1CN(C(=O)Cn2nnc(C)n2)C1)(C(C)(C)C)OC C1(C(=O)NCCNC(C(C)Sc2ccc(F)cc2)=O)CN2CCCC1C2 c1(C(N2CC(NCc3ccc(OC(F)F)cc3)C3(CC3)C2)=O)ccc(F)c(F)c1Cl c1(C(N2CCN(C(=O)NCCc3ccc(C)s3)CC2)=O)ccn2cncc2c1 c1(OC)ccc(C(C)C(=O)NCC2CCC2NC(=O)Cc2ccnn2C)c(C)c1 C1(=O)CCCCCCN1.CCCC(O)C(CO)NC(=O)CCOCCOCC N1(C(C(C)(C)F)=O)CCC2(C1)CN(C(c1cnc(O)[nH]1)=O)CCO2 C(=O)(C(COCC)N=[N+]=[N-])NCC(C)NC(C(C=C)CC)=O c1(OC)c(C(=O)NCC2CCCCC2NC(C2CCCO2)=O)cnn1C C1(C(C)C)CN(C(=O)Cc2cscn2)CCN1C(=O)C(O)Cc1cccc(Cl)c1 c1(NC(C=C(C)C)=O)ccc(-c2cn(C3C=CCCC3)nn2)cc1 Nc1ccnc2sc(C(=O)Nc3cccc(OCc4ccc(F)cc4Br)c3)cc12 N1(C(CCCC#C)=O)CCCC1C1CCCCN1C(c1cc(CC)c[nH]1)=O N1(C(CC(CC)SC)=O)CCC(NC(c2cnc(C(N)=O)cn2)=O)C(O)C1 C1(NC(Cn2c(C)nc(C)n2)=O)CN(C(C2SCCS2)=O)CC(F)(F)C1 N1(C(C=CC=CCC)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)C(C)CC1C C1(CC)CC(C(=O)NCC(O)C(C)(C)C)CCN1C(=O)CC1CCCN1C CC(C)(C)C(C(=O)NCC1=CCCOC1)NC(C1CCCN1C=O)=O C1(N(C)C(C2CCCN(C(=O)OC(C)(C)C)C2)=O)CCC(NC(=O)C=CCO)CC1 c1(C(C)C)nccc(=NCC2CN(C(=O)CC3CC(C)OC3C)CC23CCC3)[nH]1 c1(CCC(=O)CNC(=O)N)ccc(SC)cc1.C1(C(=O)OCC)CC1.C1(N)CC1 N1(C(Cn2c(C)ncc2)=O)CCOC(CCNC(=O)C(c2cnn(C)c2)=O)C1 c1(C(N2C3CN(C(C4CC(C)(C)C4)=O)C(CC3)C2)=O)ccc2cc(N)ccc2n1 c1(C(=O)NCC2CN(C(CN(C)C)=O)CC2O)cnn2c1S(=O)(=O)NCC2 Cc1ccc(C(=O)NC2C3CC4C2C4C3C(=O)NC2C(=O)N(C)CC2C)cc1O C(=O)(C1=CCCC1C)N.C1(C(=O)OC)(N(C(=O)C=CCF)C)CC1 Cc1nccc(C(=O)N(C2CCCC(NC(=O)CN3C(=O)CNC3=O)C2)C)n1 N1(C(c2cc(COC)sc2)=O)CCCC(NC(c2cccc(OC)n2)=O)C1 CC(C)C(CNC(C1(C)COC1)=O)C(=O)N(C)Cc1cccnc1 C1(C(=O)NC2CC(CNC(C=CC=CC)=O)C2)COCCN1C c1(C(N2CCC(C#C)C2)=O)cc(Cl)nc2ccccc12.C(=O)(C1=CC=NC(=O)C1)NBr c1(C(=O)NC2(CC(=O)NC(CC)C(C)O)CCC2)ccnnc1O N1(C(C(C)N(CC)CC)=O)CCC(C(=O)NC(c2nnc(C)s2)C)(CC)C1 c1(C(=O)NC2(CC=C)CN(C(C3CC(C(C)C)=NO3)=O)C2)c(C)nc(O)nc1S c1(OC)ccc(N(C(C(=O)NCc2nccs2)C2CCOC2)C)cc1C N1(C(CC=C)=O)CCC(C)(CNC(c2ccc(-c3cnn(C)c3)cc2)=O)C1 c1(C(=O)NCC(CO)NC(=O)CNC(C2CCC2)=O)cccc(C2CCOC2)c1 C(=O)(CS(=O)(=O)CC(=O)NC1CCCCC1NC(C1CCCC1O)=O)OC CCCC(C(=O)NCC1CCOC1(C)C)NC(c1ccccc1O)=O N1(C(=O)NC(CC(C)C)C)CCCSCC1C(=O)Nc1nc(C(C)(C)C)cs1 c1(C(=O)NCC(CC)NC(=O)CCc2cncs2)ccc(NC(N)=O)cc1 C#CCC(CC#C)C(=O)N(C)CCN(C)C(C1Cc2ccncc2C1)=O N1(C(c2c(CC)nco2)=O)CCC2CC2(C(=O)Nc2ccc(C)c(C#N)c2)CC1 c1(-n2cc(C(C(=O)OC)C3CC3)nn2)cccc(CC(CONC(=O)OC)C)c1 C=CC1(CC(=O)NCC2CCCC(C)O2)CN(C(c2ccc(C)s2)=O)C1 C1(NC(c2cccc(C)n2)=O)CCC2(CC1)CN(C(=O)C(C)C1CCCC1)C2 c1(CC(N2C(CCNC(c3c(C)sc(O)n3)=O)CCCC2)=O)c(F)ccnc1Cl Cc1cc(NC(=O)C(C)NC(=O)CCC2CCC(=O)C2)c(F)cc1F CCC(CC)(C(=O)N(C1CCN(C(=O)C(C)=C(C)C)C1)CCO)c1cccc(Cl)c1 c1(OC)ccnc(OC)c1C(=O)N(C)CC1CCCN1C(c1cc(O)cs1)=O C1(NC(Cc2ccn(CC)n2)=O)CN(C(c2[nH]ccc2COC)=O)CC1O c12ccnc(c1)CN(C)C2=O.Cc1occc1C(N1CCCC1C1CC1)=O CC(C)(CNC(C1(O)CC1)=O)CCNC(=O)Cc1csc(C2CC2)n1 CCC(C)(C(=O)N1CCc2sccc2C1CNC(C1(C)CC1)=O)C(F)F CCC(C)C(CC(=O)N(CCN(C)C)C(C)C)NC(C1CC12CC2)=O C1(NC(C2(CC)CCCC2O)=O)C2CCN(C(=O)C=CC(F)(F)F)CC12 N1(C(COCCC=C)=O)CCN(C(=O)C2=CCOC2)C(CF)C1 N1(C(C2CN(C)C(=O)C2)=O)CC2CCC1CN2S(=O)(=O)Cc1ccc(F)cc1F c1(CNC(C2(NC(=O)CC3(O)CCCCC3)COC2)=O)ccccc1[N+](=O)[O-] N1(C(C2(COC)COC2)=O)CCC(F)(CNC(C2CC(C)CO2)=O)CC1 Cc1nc(O)nc(C)c1C(=O)NCC1CN(C(=O)C(C)(Cl)Cl)CCC1C Cn1cc(C(N2CC(C(=O)NCCNC(=O)C=Cc3cc[nH]c3)C2)=O)c(C2CC2)n1 c1(-c2c(C)nn(C)c2)cccc2[nH]nc(C(=O)Nc3ncc(I)cc3Br)c12 c1(NC(CCSCC)C)ccc(S(=O)(=O)N2CC3OCOC3C2)c(Cl)c1 C=CC1CN(C(C2CC(CF)C2)=O)CC1NC(c1cc(Cl)cnc1C)=O C1(NC(C(=O)NCC(C(=O)OCC)C(C)C)=O)CCCc2ccccc2C1 N1(C(CC=C=C)=O)CCC(C(=O)N(CC(O)COC)C)(C(C)C)C1 C12(CCNC(C=CCOCCOC)=O)CCC1CN(C(C1(C)CC1(Cl)Cl)=O)C2 C1(NC(c2onc(CC)n2)=O)CCC2CN(C(=O)C(CCO)N(C)C)CC2C1 c1(C(N2CC(C(C)NC(=O)C(C)NC=O)OCC2)=O)cc(S(N)(=O)=O)co1 c1(OC(C)C)ccc(C(=O)NCC2(C)CCCN2C(C2CCCS2)=O)c(Cl)c1 C(C)(C)(C(C)CC(=O)N(C(C)CN(C)C(C)=O)C)NC(CC(CC)O)=O c1(-c2cn(CC(N3C(C)CC3C(N3CC(CO)C3)=O)=O)nn2)ccc(Cl)cc1Cl C1(NC(C2CC2(C)C)=O)CCN(CCSc2cn(CSc3ccccc3)nn2)C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)Cc2ccc(OC)cc2)ccc(C)nc1 c1(C(CCC(=O)N(C(CC)CNC(C)CC(C)C)C)=O)cc2n(n1)CCNC2=O c1(C(=O)NC(CC)CNC(C2CC23CC(C)(C)C3)=O)cc(Cl)cc(F)c1F N1(C(c2cc(OCC)c(C)cc2)=O)CCC2(CCC2NC(C2CC2(F)F)=O)CC1 N1(C(C(C)OC2CCOC2)=O)CC2CC1C2NC(=O)C(C)c1ccco1 N12CC(C3(CCCCC3)C1)C(=O)C(=O)CCNC(=O)C2C1CC1(C)Br.CCO.OC c1(CCCSCC)nc(-c2ccnc(C(F)(F)F)n2)n(-c2ccnc(Cl)c2)n1 CN1N=CC(CC(N2CCC(C(N3CCSCC3)=O)(CO)C2)=O)C1=O C1(C(=O)NCCN(CC(C)O)C(c2c(C)nsc2)=O)CCCN(C(N)=O)C1 C1(CN(C(=O)Cc2ccccc2)C)CC(F)CN1C(C1CCC(C(N)=O)CC1)=O c1(C(N2CCCC(N(C(c3cc(C)sc3C)=O)CCF)C2)=O)ncn2c1CCC2 C1(NC(Cc2scc(C)n2)=O)CCCCC12CCN(C(=O)C(=O)C(F)(F)F)CC2 Cc1nn(C)cc1-c1cn(CC(F)CCNC(=O)CC2COC(C)(C)C2)nn1 N1(C(C(CCC)OC)=O)CC(CNC(c2c[nH]nc2[N+](=O)[O-])=O)CC1(C)C N#Cc1ccccc1OCC(N1CCCCC(NC(C2(CO)CC2)=O)C1)=O N1(C(C2(OC)CCC2)=O)CC2CCC2(C(=O)NCC(O)CC2CCCC2)C1 c1(C(C)NC(=O)CCNS(C)(=O)=O)cccnc1O.C12CCC(C1)NC2=O C12(C(N3CC(C)C(F)C3)=O)CCC(NC(c3cncnc3)=O)(CC1)CC2 c1(OCCCN(C)C)ccc(NCC(c2cccnc2)O)cc1 C1(NC(c2cc(CC)no2)=O)CC2(CCN(C(C34CCCC3CCC4)=O)C2)C1 N1(C(CCN(CC)CC)=O)CC2CC(NC(c3ccc(Cl)c(Cl)c3)=O)C2C1 N1(C(C2C(CN(C)C)C2)=O)CCC(CNC(C2CC(F)(CN(C)C)C2)=O)(CO)C1 CC(C(=O)Nc1ccc(C(N)=O)cc1)S(N)(=O)=O.C12(CO)C3CC(CC13)C2OC c1(SCC)ccccc1C(=O)NC12CC(CNC(=O)COC3CC(F)(F)C3)(C1)C2 C1(CNC(c2ccc(F)c(F)c2)=O)CCCCCN1C(=O)C(CO)c1ccccc1 CC(CS(C)(=O)=O)C(=O)N1CC2(NC(=O)Cn3cc4ccccc4n3)CCC1C2 c1(CC)cccc(C(=O)NC2CC2C(=O)N(C2CC2)Cc2ccc(C)cc2)c1 c1(C(C(=O)NCC=CCNC(CC(c2ccccc2F)C)=O)O)cccc(F)c1 O=C(CC1=CCCC1)N1CC2C(C(=O)NCCCF)C2C1 N#CC1(C(N2CC3(CCN3C(=O)CN3CCN(C4CC4)CC3)C2)=O)CCCOC1 NS(=O)(=O)c1ccc(C(=O)NCC2CC(NC(c3cscc3F)=O)C2)cc1 C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CCNC(c2c(C)cnnc2)=O)CCC1 c1(CN(C(=O)CC2CCN2C(C2CC=CC2)=O)CC)cnn(C)c1 Cn1nc(C(C)(C)C)cc1CNC(C1(C(=O)O)CC(F)(F)C1)=O CN1CCOC(C(=O)NC2(C(=O)N(C3CC(F)(F)C3)C)CCOCC2)C1 C1(C(N(C(C2Cc3ccccc3O2)C)C)=O)Cc2cccnc2NC1=O N1(C(CCNC(C)=O)=O)CC2CCC1CC2NC(c1ccnc(CO)c1)=O CC(C(C)(C)C(=O)N1CCCCCC1C)NC(c1ccccc1C1CC1)=O C12(CC(=O)NC3CCC(NC(C(C)Cc4ccccc4)=O)C3)COC(CF)(C1)C2 C1(CC)CCN(C(=O)Nc2cccc(C(=O)NC(N)=O)c2)CC1(F)F C#Cc1ccc(C(=O)NCCC2CCCN2C(=O)C(CC)NC(N)=O)c(F)c1 N1(C(Cc2nc(C)oc2)=O)CC2=C(C1)CN(C(c1nnn(C(C)(C)C)n1)=O)C2 C=C(C)C(CC(=O)N(CC(C)O)CCNC(c1cc2occc2s1)=O)OCC C1(C(N2CCN(C(CCC)=O)CC2)=O)CC12CCN(Cc1nc(Cl)ccc1F)C2 C(=O)(CC(C(F)(F)F)OC)N1CCC(N(C(=O)C(=CC2CCCCC2)F)CC)C1 C1(C(N2CC3CC2C2CC32)=O)C2CCCC2CN1C(c1cn(C2CC2)cn1)=O c1(C(N2CCC(O)(CC(=O)NCC3CCCO3)CC2)=O)ccc(Cl)c([N+](=O)[O-])c1 C1(CNC(c2ccc(C(F)F)o2)=O)C2CN(C(=O)C(c3ccc(O)cc3)=O)CC12 CC1CCC(NC(C2CC2C)=O)CN1C(=O)Cn1nc(C(F)(F)F)cc1C(F)F C1(CC(=O)NCC(CNC(c2c(C)cc(SC)o2)=O)C)COc2ccccc2O1 C1(N(C(=O)C(F)=CCCF)C)CCC(C(N2CCC(C(C)O)C2)=O)CC1 N1(C(C(C)CSC(F)(F)F)=O)CCN(C(c2cn(C)nn2)=O)C(c2cn[nH]c2)C1 O=C(C1CCCn2ccnc21)NC1(CNC(C2C3CCCCCCC23)=O)CC1 Cc1ncn2ccc(C(N3CC4C(NC(c5nn[nH]c5Cl)=O)C4C3)=O)cc12 C1(C(=O)NC2CC3(CC(NC(C(C4CC4)SC)=O)C3)C2)CCc2nn(C)cc2C1 C1(C(=O)NCC(CC)NC(c2c[nH]nc2CN)=O)CCCC(N(C)C)C1 N1(C(=O)CC2(CO)CC2)CCC2(C1)CN(C(c1ccnc(O)c1Br)=O)C2 c1(N2CC(C#N)OCC2)nc(=NCc2nnnn2C)[nH]c2c1SCC2 C(=O)(CC(C)(C)CC(F)(F)F)N(CCCNC(=O)Cc1ncc(F)cc1F)C N1(C(c2cnn(CCCC)c2C)=O)CCC(CNC(c2cc(Cl)on2)=O)C12CC2 N1(C(CC2N(C(c3ccc(SCC)nc3)=O)CCC2)=O)CC(OC)CCC1C c1(CC(=O)NC2CCN(C(C3C(C)(C)OCC3)=O)C2(C)C)cn2c(n1)CCCC2 N(C(=NCC(=O)Nc1cccnc1)NC1CCCC1)C(C1CCCC1)C#C C1(O)(CNC(c2cccc(OC)n2)=O)CCN(C(c2ccc(=O)n(C)n2)=O)CC1 N1(C(c2c(CC)nns2)=O)CC2(C1)SCCC2NC(C1CC=CCO1)=O N1(C(Cn2c(C)ccn2)=O)CCC2(CC(C(=O)N(C)CCC3CN(C)C3)C2)C1 N1(C(CCS(N)(=O)=O)=O)CCCCCC(NC(c2cc3cc(Cl)sc3[nH]2)=O)C1 N1(C(CCNC(C)=O)=O)CCCCC1CCCNC(C1(C(F)(F)F)CCCCO1)=O CC(C)CC(CC(=O)O)NC(=O)C(C)Cc1cn(CCC2CCCN(C)C2)nn1 c1(OC)ccc(C=CC(=O)NC23CCC(C2)N(CC2CCCO2)C3)nc1 C=C1CC2(C1)CC(C(=O)NCc1csc(CNC(=O)CCC(F)(F)F)n1)C2 c1(C(=O)OC)c[nH]c(=NCCCCC(C)NC(=O)C(C)C(C)C)cc1C N1(C(C(C)OCCC=C)=O)CCCCC(N(C)C(c2ccc(CSC)cc2)=O)C1 c1(C2(SC(NOC(C)(C)C)=O)CC2)cn(CCNC(=O)CNC(N)=O)nn1 C(C1CCS(=O)(=O)c2ccccc21)NC(C(=O)NC1CC(C(C)(C)C)OCC1)=O Cc1cc(C(=O)NCC(C)(C)CC(=O)NCCC2(O)CCOC2)cnc1C O(P(=O)(CCC(C)(C)C)C(=O)N(CC(F)(F)F)C)CC(CCC)Cl C1(CC)C(NC(=O)Cn2cncn2)CCN1C(c1cc(C(C)C)nn1C)=O c1(C2(NC(CN3CC(C)C(C)C3)=O)CCC2)c(F)cccc1F O=C1CC2CC(C(N3CCN(C(=O)CCc4ncco4)CC3)=O)C1C2 C(c1cc(F)cc(F)c1)=CC(N1CC2C(NC(C3(CO)CCC3)=O)C2C1)=O N(C(=NCC1CCOC1)N1CCC(C2CCC2)C1)Cc1cc(CC)no1 Cc1cccc(F)c1C(=O)NCCC1(NC(=O)CC2CCCNC2=O)CCC1 c1(N2CCC(C(=O)NCCCc3c(C)cccc3)CC2)ccccc1[N+](=O)[O-] C12(CN3CC(CCC)OCC3)CCC(C1)C(=O)NC2 c1(C(=O)NCC2C(Cn3cc(CN(C4CCCC4)C(C)=O)nn3)C2)[nH]c(O)nc1C c1(C(=O)NC2CC(CC(=O)NC3C(CN=[N+]=[N-])CCC3)C2)cncc2[nH]ccc12 N1(C(CNC=O)=O)CCC(C(F)(F)F)CC1CNC(c1cc(C(N)=O)[nH]n1)=O N#Cc1ccnc(NCCN(C(C2CC2C2CCCO2)=O)CC2CC2)n1 C#Cc1cc(C(=O)OC2CCN(CCO)CC2)ccc1Cl c1(C(=O)NC(CNC(CC(C=C)C)=O)C2CC2)ccc(OC)c(OC)c1C N1(C(C(CN(C)C)NC(C(C)OCC)=O)=O)CC(C)(C)CC1C CC1(NC(=O)Nc2cccc(-c3ncc[nH]3)c2)CCOC1C1CC1 CC1CCN(C(=O)CCc2ccccc2F)C1CNC(c1ccc(N)cn1)=O N1(C(C=CC)=O)CCC(C2CCN(C(=O)Cc3nc([N+](=O)[O-])n[nH]3)CC2)C1 N1(C(C2(NC(c3n(C=C)nnc3)=O)CCOCC2)=O)CC(O)C(C)(C)C1 c1(C2(C(N(C3CCN(C(C(C)OCC)=O)CC3)CC)=O)CC2)ccc(F)c(F)c1 C1(n2cc(CC(C)C)nn2)CC2(C1)CC(C(=O)NC1COCC1N=[N+]=[N-])C2 CCC(C)C(=O)C(=O)NCC(C)NC(c1nnnc(O)c1C)=O c1(C(=O)NC(CCNC(CCCOCCOC)=O)C)cc2c(C)ccc(C)c2[nH]1 C(COCC)(C(=O)OC)NC(=O)CSc1cccnc1.C1C(=O)N1CCC C1(CC(=O)N(CC#C)C)CC(F)(F)CN1C(=O)C(C)CSC N1(C(C23CN(C(C(CCOC)C)=O)C(C2)CO3)=O)CC2CCCCC2C1 C1(NC(c2c(OCC)ccs2)=O)CCC2(C1)CN(C(c1cc(F)c(Cl)cc1F)=O)C2 C1(C(=O)NCC(O)C(F)F)CCCCCN1C(C1CC2CCC(C1)O2)=O CCCC(CCC)C(=O)NC1CCC(NC(c2cc(C3CCC3)no2)=O)C1 c1(C(=O)NCCN(CCC)C(C2CCCC23CC3)=O)cc2c(C)cc(F)cc2[nH]1 C(c1c(F)cccc1F)=CC(=O)NC1CCCC(NC(CCC(C)(F)F)=O)C1 CCCCC(C)N=c1cc(C)[nH]c(=NCC(C)CCCN2CCOCC2)[nH]1 S(=O)(=O)(c1ccc(Cl)c(C#N)c1)N1CCC2(C(=O)OC(C)(C)C)C(C1)C2 C(=O)(C(C)C=C=C)N1C(CC(=O)NCCOCC#C)CCC1 CCC(C(=O)N1CC(CNC(=O)CSc2n[nH]c(O)n2)C(C)C1)C(C)C N(C(=S)c1ccccc1)(C(c1ccc2[nH]c(C(F)(F)F)nc2c1)=O)CC C=Cn1nccc1C(=O)N(C(C)CNC(c1sc(-c2ncc[nH]2)nc1C)=O)C c1(C(N(CC(CNC(c2nc(CC)oc2)=O)O)C)=O)cccc(C2COC2)c1 N1(C(CCN(C)CC)=O)CCCCC1C1CCCN1C(c1ccc(=O)oc1)=O C=CCC(CC=C)C(=O)N(CCCCN(C)C(C1CC2(C1)CS(=O)(=O)C2)=O)C c1(CC(=O)OC)cccc(C)c1.CCC(=O)NC1CC1.C(CCNC(=O)N)NCC c1(C(=O)NCC(=O)NC(CC(C)NC(C2(CC)CCC2)=O)C)cncc(Br)c1 N1(C(c2cnc[nH]2)=O)CCC2(CCCN(C(C3CC34CCCCC4)=O)C2)C1 CC(C)C(CCC(=O)N1CCN(C2CCC2)CC1)NC(=O)CN1CCCC1C C1(C(=O)NC(=O)C=CC2CC2)CCC(OC(C2CC2Oc2ccccc2)=O)CC1 C1(CC(=O)NCCC2(O)CN(C(C3C(C)C3)=O)C2)CCC(=O)N1C N1(C(C(C)=CC)=O)CC(CNC(=O)CCOCCCOC)CC1(C)C C1(C(=O)NC(C2CN(C(=O)CN3CC4CC4C3)C2)C)CCS(=O)(=O)N1 N1(C(c2n(C)cnc2)=O)CCC2(COCC(CNC(c3cccnc3S)=O)O2)C1 CCCC(C)CC(=O)N1CC=CC(NC(c2ccn(C3CCOCC3)n2)=O)C1 C1(O)(C(=O)NC(c2ccoc2)C)CCN(C(=O)Cc2ccc(Br)cc2)CC1 n1(CC(N2CC(C3(NC(C4C(C)CCO4)=O)CC3)C2)=O)nc2c(n1)CCCC2 N1(C(=O)NC(C)(C)C(F)(F)F)CCCC(C)(C(=O)Nc2cnc(Cl)nc2)C1 c1(C(=O)NCC(C2CCOC2)NC(c2c(C)[nH]nc2Cl)=O)csc2c1CCCC2 C1(C)COCCC1c1nc(C(c2ccccc2Br)(F)F)nn1-n1c(C)ncc1 C1(NC(c2oc(C)c(CO)c2)=O)CCC(C(=O)N2CCn3nccc3C2)=CC1 c1(C(=O)NC(CNC(c2ccc(F)c(F)c2F)=O)CO)ccc(F)c2c1OCC2 C1(NC(CNC(CC)=O)=O)CCCC12CCN(C(=O)CNC(C)=O)C2 C(=O)(C1=CCC2CCC1N2C(=O)CC(C)SC)N(CC(CC)O)C C1(CC)(NC(C2CCCCC2(C)C)=O)CCN(C(=O)C(C2CCCCC2)O)CC1 Cc1cccc(F)c1C(=O)NCC(O)CNC(c1csc(CS(C)(=O)=O)n1)=O Cc1ccc(C(=O)NCC2CCN2C(C2CC3(CCC3)CO2)=O)c(O)c1 C(c1cocn1)=CC(=O)NC1CCC(NC(=O)COCc2nc[nH]n2)C1 C(=O)(C(C(C)NC(C1CC2CC(=O)C1O2)=O)C(C)C)NCC=CCCC c1(OC)cc(NC(=O)C(CC(C)C)OC)cc(C(=O)NNc2cccs2)c1 c1(NC(C2C(CNC(C(C(COC)C)C)=O)CCCC2)=O)ccc2nncn2c1 c1(C(N2CCC(N(C(=O)CC(C)F)CC)C2)=O)ccnc(C)c1C CS(=O)(=O)c1ccc(C(=O)NC2CN(C(C3CC3C#N)=O)C3(CCC3)C2)s1 C1(C(=O)NC2(CNC(c3scc(OC)c3)=O)CC2)OCC2CCCCC12 C(=O)(CCCC(F)(F)F)N1CC(CN(C)C(c2cc(F)cc(F)c2)=O)OCC1 CC1(CNC(C2(C(F)F)CCCC2)=O)CCN(C(c2cc(O)cs2)=O)CC1 N1(C(C2C(OC)CCC2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1CO N1(C(C(C(=O)OC)C)=O)CC2(C1)CN(C(C1(n3nccn3)CC1)=O)C2 c1(C(N(CCCNC(C2CCCO2)=O)CC)=O)cccc(C(F)F)c1F c1(C(=O)NC2CC(NC(c3c(CC)cno3)=O)C23CCC3)n[nH]c(C)c1[N+](=O)[O-] C1(C2CC2)(NC(CCC=C=C)=O)CCN(C(=O)CCOc2ccccc2C)C1 c1(C(N(C2CCN(C(C3COCC(C)(C)O3)=O)C2)CC)=O)cc(C)ccc1F c1(C(CCC)[SH](CCC#C)C)ccc(C#N)cc1 C1(C(=O)NCc2cc(C(N(CC(COC)(C)C)C)=O)n(C)n2)CCCC2(CC2)C1 C(CCC(O)C(=O)NC1(C(C)C)CC1)NC(C1C(CC)C1)=O n1(CCCC)cc(C2(C(=O)OC)CN(C(=O)C(n3cc(Br)cn3)C)C2)nn1 c1(C(N2CCCC(CCNC(CC)=O)C2)=O)cc(O)cc(O)n1 C1(NC(C=C(CCN(C)C)Cl)=O)CCN(C(C2CCCC3(CC3)C2)=O)CC1(C)C C12(C(=O)NCC(C)(C)NC(C3CCC4(CC3)CC4)=O)CC3CC(C1)CC(O)(C3)C2 CC1CCC(=CC(=O)NCCCCN(C)C(c2n[nH]cc2C2CC2)=O)CC1 C(=O)(CC(C)P(C)(C)=O)N1C(CO)CC(NC(c2c(CC)ocn2)=O)C1 N1(C(C2(CC(C)C)CC2)=O)CC(N(C)C(C2CC(=C3CC3)C2)=O)C(O)C1 C(C(=O)N1CC(NC(=O)CC2OCCCO2)C1)(C(C)C)NC(C(C)OC)=O N1(C(c2c(CC)nn(C)c2)=O)CC2(CCC2NC(=O)C(C)SC(C)C)C1 N1(C(C2(C(=O)NC)CCC2)=O)CCCN(C(C2CCC(=O)NC2)=O)C(C)C1 c1(CC)cnc(O)c(C(=O)NCC2CCN2C(c2cc(Cl)cnn2)=O)c1 c1(N(C(c2cncs2)C(=O)N)OCC)ccc(F)cc1.C1(C)CCCO1 C1(CC)C(C(=O)NOCCOC(C)=O)CCCN1C(c1ncc(N)cc1C)=O c1(C(=O)NC(C2CCCCC2)CNC(=O)CCc2cc(Cl)no2)cc2sccc2[nH]1 C(=O)(C1=CC(C)(C)C1)NCC1(NC(=O)CC2CCCOCC2)CC(OC)C1 c1(CCNC(=NC)NCCc2csc(-c3nnc(CC)o3)n2)ccccc1Cl CCC(C)C(C(=O)NC(C)(C)CCCNC(c1cccc(Cl)c1OC)=O)OC N1(C(CC2CC(OCC)C2)=O)CC(O)CC1CNC(c1cc(C)oc1CC)=O C1(C)(CC)CCCN(C(=O)C(O)C2CN(C(=O)Cc3csnn3)C2)C1 CC1(C)CN(C(C2CC(F)(F)C2)=O)C(CNC(C2CCS(=O)(=O)N2)=O)CO1 CN1CCCC(NC(=O)C(Cc2ccco2)NC(c2ccc(C#N)n2C)=O)C1=O Nc1c(C(=O)NC2CCCCC2NC(C2C3CCC(=O)C23)=O)ccc(F)c1F c1(NC(=O)NCc2cc(C)c(I)cc2)ccc2c(c1)CC(N)C2 C1(O)(C(=O)NCCSCC(=O)NCC2(C(C)(C)O)CC2)CCCC1 c1(NC(C)=O)cccnc1C(=O)NCC1(C(=O)NCC2CCC=CO2)CCCO1 C#CCCCC(=O)NC12CC1CN(C(=O)C(C)(F)c1ccccc1)C2 c1(C(N2C(CNC(C3N(CC)CC3)=O)C=CC2)=O)ccc(C(F)(F)F)c(F)c1C N1(C(C(=O)NC(CC)(C)C)c2cccs2)CCc2c(F)ccc(C#N)c2C1 c1(C(=O)NC2(C)CCN(C(CC3C(C)(C)C3)=O)C2)cc(Cl)cc2c1OCC2 C1(C(=O)NCc2cc(C(C)C)no2)CCCCC1NC(=O)Cn1ncnn1 c1(C(=O)NCC2N(C(Cc3c(C)occ3)=O)CCC2C)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC(NC(c3n(CC)nnc3)=O)C(CO)CC2)=O)cnn2ccn(C)c12 CC1CN(C(=O)C(F)Br)CC1n1cc(-c2ccsc2)nn1 C=CC(C)(CCOC)C(=O)N1CCN(C)C(C(=O)NCC2CCCN(C)C2=O)C1 C1(CCNC(C)C(N)CC(F)(F)F)CC(C)(C)OC(C)(C)C1 C(C)(C(=O)NCCSCC)NC(CSCC#C)=O n1(CC(=O)NC2(C)CCN(c3ncc4ncnc-4[nH]3)CC2)ncc2cccnc12 C(C(COC)N=c1nc(CSC)cc(C)[nH]1)NC(CS(CC)(=O)=O)=O N1(C(=O)CSc2ncccc2F)CC(NC(=O)CCc2cncs2)C(F)C1 N1(CC)CCOCC1C(=O)NC(C)CCCCNC(=O)CCn1c(C)ccc1C C1(NC(=O)CCn2ccnc2)CC2CC1CN(C(c1cccc(F)c1F)=O)C2 c1(C(=O)NC2(COC)CCN(C(=O)CCc3ncccn3)C2)cc(F)ccc1Cl N#Cc1ccccc1OCCS(=O)(=O)NCC(=O)Nc1cccc(F)c1 c1(NC(CCN2CCC(CCCCC(=O)OCC)CC2)=O)ccc(Cl)c(F)c1 CCCC(C)CC(=O)N1CCC(CCC(=O)NC23CC2CN(C)C3)C1 C1(O)(C(CNC(CCSC)=O)(C)C)CN(C(c2coc(N(C)C)n2)=O)C1 C1(NC(C(CC)C(C)(F)F)=O)COC2(CCN(C(=O)C(C)C)CC2)C1 CCC(CC(=O)N1CCC(C)(C)C1C(=O)N(C)Cc1sccc1C)CC(C)C C1(C)(C(=O)NCC(C2CC2)NC(c2ccn(CCOC)n2)=O)CC(C)=NO1 C(=O)(CCCC(C)(C)C#N)NC1C(C(N(CC(CC)O)CC)=O)CC1 C#CC1(C(=O)NCC(O)CC(=O)NCC(C)C(C)C)CCCCC1 CCCCCC(O)CC(=O)N(C(C)C(N1CC(C)(C)CC1C)=O)CC CCS(=O)(=O)CC(=O)N1CC2CC(NC(c3cncc(C)c3Cl)=O)C1C2 N1(C(C2(CCCC)CCCC2)=O)CC(NC(=O)C(C)(C)CF)C(F)C1 C(=O)(CCC(F)(F)C(F)F)NC(C(C)NC(c1nc(CCC)sc1)=O)(C)C Cc1cc(=O)ccn1CC(=O)NCC1CC1CNC(c1cncc(C#N)c1)=O c1(C(=O)Nc2ncccc2F)ccc(Cl)cc1Cl.C1CCN1.C(COC)O Cc1cc(NC(=O)Cc2cccc(CNC(c3ccco3)C)c2)n(C)n1 Cc1csc(C(C)C(=O)N(CCNC(C2COC(=O)N2)=O)C2CC2)n1 N1(C(C(CNC(=O)Cc2csc(C)c2)OC)=O)CCCCC1C1CC1NC(C)=O c1(C(N(CCCN(C(C(C)Oc2cccc(F)c2)=O)C)C)=O)cncc(F)c1Cl CCC(F)(F)C(C)(C)C(=O)NCCC1(C)CCN(C(=O)C(C2CC2)OC)CC1 N1(C(C(CC)=CCCC)=O)CC(C(=O)Nc2ccc(N(C)C)nc2)CC(C)(C)C1 c1(C(=O)NCCNC(=O)CSC2CC3CCC2C3)cccc(N2CCOCC2)c1 C1(CNC(C(C)=C2CC2)=O)(CNC(c2ccnn2C2CC2(F)F)=O)CC1(F)F N1(C(C(=O)NC2CC2)=O)CCC2CN(C(=O)CC3OCCCO3)CC12 c1(NC(N2CC3(CCCCCC3)C2)=O)nnc2n1CCCCC2 c1(C(N(CCCNC(CNC(CCC)=O)=O)C2CC2)=O)sc(O)nc1C C1(NC(=O)Cc2cc[nH]c2)CC2(CCN(C(=O)Cc3ccsc3Cl)C2)C1 c1(SC)ccccc1CC(=O)N(CCCCNC(C1CC1(F)Cl)=O)C c1(C(=O)NC(CN(C(=O)Cc2occc2C)CC)C)nccn2nccc12 c1(C(=O)NCC(C2CC2)NC(C(N2CCCCC2)C)=O)occ2c1CCC2 N1(C(C2CC(=O)C23CCCC3)=O)CCOC2CCN(C(C3(F)CCCC3)=O)CC12 Cc1cc2ncn(CC(=O)NC3CC(O)CN(C(C4CC(O)C4)=O)C3)c2cc1C c1(C(=O)NCc2c(OCC)c(Cl)ncc2)cc(F)ccc1C(C)C C=C1CC2(C1)CN(C(=O)CC1CN(C(c3ccc(C#N)cn3)=O)CCC1C)C2 c1(C(=O)NC(C(C)NC(CCc2cc(C)no2)=O)C)ccc(-c2ccsc2)cc1 N1(C(Cc2nc(C)[nH]n2)=O)CC2CCCC1(CNC(C1CCCCC1O)=O)C2 c1(CNC2CC(NC(c3c(F)cc(O)cc3F)=O)C2)cccc2nccnc12 CC1CN(CC2COC(C)(C)O2)CCC1NCc1cnc(-c2ccccc2)[nH]1 c1(CC)ccc(S(C)(=O)=NC(=O)CC(C)(C)OC)cc1.C1(C)(C)C(=O)N1 C1(C(N(C)CCOCCNC(c2ccc(CF)cc2)=O)=O)CCc2cncn2C1 CC1(C)CCC(NCc2nnn(-c3ccc(C4CCC4)cn3)n2)c2ccccc21 c1(NC(C2C3CC(NC(=O)OC(C)(C)C)CC32)=O)ccc2c(c1)CC(C)O2.OC N1(C(C(Cc2cn[nH]c2)NC(=O)CC=C(Cl)Cl)=O)CCC(C2CCC2)C1 C1(c2cn(C)nc2)CN(C(c2c[nH]nc2C(F)F)=O)CCN1C(C1CC12CC2)=O C1(NC(C23CC(C)C2C3)=O)CCC2(CC1)CN(C(C1(N3CCCC3)CCC1)=O)C2 c1(C(=O)NC23C(CN(C(c4ccc(C)o4)=O)C2)C3)cc2sc(C)cc2s1 C(=O)(C1=C(C)OCCS1)N1CCC(C=C)(C(N2CCOCCC2C)=O)C1 c1(C(N2C(C)CC(NC(C=COCC)=O)C2)=O)cc(Cl)ccc1Cl C(=O)(CCCCCCN=[N+]=[N-])N1C(CNC(=O)CCC2CCCO2)CC(OC)C1 c1(CC)ccc(-c2nc(-c3cnc(-c4ccccc4)nc3)no2)cc1 c1(-c2cn(CC(C)OCc3c(C)c(C(C)C)no3)nn2)ccc(=O)n(C2CC2)c1 Cn1cc([N+](=O)[O-])c(C(=O)NC2CCCN(C(=O)Cc3ccns3)CC2)n1 C(=O)(CCCN=[N+]=[N-])NCC1(CNC(C2C(C)(C)CCC2)=O)CC1(F)F Cc1ccc2c(ccn2CC(N2CC3CCC2CC3O)=O)c1 c1(C2N(C(c3cc(F)ccn3)C(=O)NCC=C)CC(O)C2)ccc(Cl)cc1Cl N1(C(CCc2cc(C)[nH]n2)=O)CCOC(C(N2CC(OCCF)C2)=O)C1 N1(C(C(CCCC(C)C)NC(C(C)OCCOCC)=O)=O)CC(F)(C2CC2)C1 c1(C(N2CC(C)C(CNC(=O)CO)C2)=O)ccc(O)cc1F CC1(C)CC(C(C2CC2)NC(=O)N(C2CCOC2)C2CCC2)C1 C(=O)(C(C)C(O)CCCC)N1CC2CCN(C(C3N(CC)CC3)=O)CC21 C1(C(N(CCNC(=O)CCc2cc(Cl)cs2)CC2CC2)=O)Cc2nccnc2C1 C1(CNC(c2ccc(F)cc2Cl)=O)C(O)C(O)CN1C(C1CC2C=CC1O2)=O S(=O)(=O)(c1ccc(N2CSC(C)C2)cc1Br)NCC(CC(=O)NC)C C(=O)(CCC(CC)NC(c1cc(CCO)on1)=O)NC(CC#C)CO C1(O)(C(=O)OCC)CCN(C(CCCNC(C)=O)Cc2ccccc2)CC1 O=C(CC1=CCCCC1)NCCC12CCC1CN(C(C1CN(C3CCC3)C1)=O)C2 CCCCC(C(=O)NC(CNC(c1occ2c1CCOC2)=O)C1CC1)C(C)C C1(NC(c2c(SCC)nccn2)=O)CN(C(=O)CCOCC(F)(F)F)CC1(C)C C12(NC(C3C(SC)CCC3)=O)CC(C1)N(C(=O)COCc1cc(C)on1)C2 c12cc(c(C)o1)C(=O)NC2.c1(CC)ccoc1C(=O)NCC(F)Br c1(CC(=O)NCC2(C)CC(NC(C3CSCCS3)=O)C2)c(Cl)cccc1Cl C1(NC(C2CC(NC(CC3(C)CCC3)=O)C2)=O)C(=O)OCC1(C)C C(=O)(C(O)C(F)(F)c1ccccc1)NC1C(C)CN(C(=O)C=Cc2cocn2)C1 N1(C(C(C)OCC2CC2)=O)CC2CN(C(=O)C(C)(C)n3cccn3)CC2(C)C1 C(C(CC(C)C)C(=O)NOCC(N1C2CCC(C2)C1CO)=O)OC N1(CC)CC(CNC(=O)C(CC2CCCC2)NC(=O)CC(Cl)Cl)CC1=O c1(C(N2CCC(C(=O)NC(CC=C)CC3CC3)(CC)CC2)=O)c[nH]c2ncccc12 c1(C(=O)NCCC2N(C(CC(C=C)(C)O)=O)CCC2)cc2cnn(C)c2s1 C(=O)(CC(C)C(C)C(C)C)N1CCC(C(C)NC(C(CC=C)C)=O)CC1 N1(C(COCCN(C)C)=O)C2CCCC1CN(C(=O)CCCCC1CC1)CC2 c1(C(N(CCNC(c2cncnc2C)=O)CC)=O)cccc2c3c([nH]c12)CCC3 Cc1nn(CC(N2CCC(NC(c3ncccc3Cl)=O)C(F)C2)=O)cc1[N+](=O)[O-] c1(C(c2ccsc2C(=O)NCC2COC(CSC3CC3)C2)=O)c(O)ccnc1F.CO CC1c2ccc(Br)cc2OC1CNC(=O)C=C1CCN(C)C1 C1(NC(C(CCC)CCC)=O)CC1C1CCCN(C(=O)CCCOC(C)C)C1 CN1CCCCCC1C(N1CCC(CC(N2CCOC(C(N)=O)C2)=O)C1(C)C)=O c1(CNC(CCC)CC(=O)N(CC(C)CC(F)(F)F)C2CC2)ccc2n[nH]cc2c1 c1(COC)ccccc1C(=O)N(CCC(C(C)C)NC(=O)CC1(O)CC1)C C12(CC(C)(C)C1)C(=O)NC(C)C(=O)NC2.C1(OC(C)=O)(CN(C)C)CC1 C1(C(N2C(CNC(c3c(C)n(CC4CC4)cc3)=O)CC2)=O)CCCC1S(C)(=O)=O c1(CC(=O)NC2(CNC(=O)CCCc3ccccc3)CC2)cc(Cl)ccc1O c1(OC)ccc(C(C)C(=O)NCCCN(CCO)C(c2ccoc2C)=O)cc1F N1(C(CC2C(C)(C)C(O)C2)=O)CC(CO)C2(C1)CN(C(c1cc3n(n1)CCC3)=O)C2 C1(CNC(c2cnc(CC)nc2C)=O)CN(C(C2CC2F)=O)C2(CCOCC2)C1 N1(C(C2N(C(C(CC)CN(C)C)=O)CC(=O)C2)=O)CC2COCC2C1 c1(C(N(CC(CNC(C(CSC)C)=O)O)C)=O)occ2c1CCCC2 c1(OCCC(=O)N2CCC2)cccc(F)c1F.C12CCCN(CC1)C(=O)CO2 CN1CCc2ccc(C(=O)Oc3ccccc3OCCCC(F)(F)F)cc2C1 C1(CNC(C(C)=CC)=O)CC2CCC1N2C(C1CCCN(S(C)(=O)=O)C1)=O C1(CC)CC(C)N(C(c2scc(C(=O)OC)c2Cl)C(=O)NCCC2CC2)C1 C(C)(C(=O)OC)N(CCCC(F)F)CC.C(C)(CCC)N(C(=O)C[SH2]C)CCC c1(CCNC(=O)NCC2CC(C3CC3)=NO2)cc(F)c(Br)cc1F c1(C(N2CCC(NC(=O)CC3CC4(CC4)C3)(CO)C2)=O)ccc(O)c([N+](=O)[O-])c1 c1(OC)c(Br)ccc(F)c1S(=O)(=O)NCC1(F)CCOC1 CCC(CC(=O)N1CCN(CCC2CCN(C(c3ccccc3)=O)C2)CC1)OC C1(C(=O)NCC(C)CNC(C2CC(=O)N(C3CCCC3)C2)=O)CCCN1N=O N1(C(CC(C)O)=O)CC(N(C)C)C(CNC(c2csc(Cl)c2)=O)C1 c1(C(=O)NCCNC(c2cc(Cl)cnn2)=O)cc(F)c(F)cc1O CCCCCC(C)(C)C(=O)NCC(=O)NCCC1CCCS1 C(=O)(C#CC(C)(C)C)N1C(C(=O)NC2(c3ncc(C)o3)CC2)(COC)C=CC1 N1(C(C2(CC(C)C)CCCC2)=O)CCOC(C(C)NC(c2cccnc2)=O)C1 C1(NC(c2ccc(-c3cscn3)nc2)=O)CC2CC(NC(c3cccs3)=O)C1C2 Cc1cccc2c(C(=O)NC3CCCC3NC(=O)CC=C(Cl)Cl)n[nH]c12 Cc1[nH]ccc(=NC(=O)C2CCC(CNC(=O)CNc3ccccc3)CC2)c1F C1(CNC(c2c(C)nsc2)=O)CC2CN(C(=O)CCc3ccc[nH]3)CC12 C1(OCC)CC2CN(C(=O)CC(C)(C)N(C)C(c3cc(=O)cc[nH]3)=O)CC12 Fc1ccc(Cl)c(I)c1C(N1CCCC1C1CCCOC1)C1CC1 CC1NC(=O)CCC1CNC(=O)CC1C2CCCC2N1C(c1cc(CO)on1)=O C1(NC(CC(=C)Br)=O)CCC(CNC(=O)CN2CCCC2=O)CC1 C1(NC(C2CC(NC(C3CCCN(C)C3)=O)C2)=O)CC12CCCCC2 CC1=CCC(C(N2CC=CC(NC(=O)CN3CCCC3=O)C2)=O)CC1 c1(C(N2CC(NC(CSC)=O)C3C2C3)=O)ccc(OC(F)(F)F)cc1O c1(C(c2n(CCC)nnn2)NCCc2cccc(Cl)c2F)cc(Br)ccc1F c1(Cc2cn(CCNC(C(C(C)O)NC(=O)C3CC3)=O)nn2)cc(F)cc(F)c1 C(=O)(CCC1=CCCCC1)N(C(C)C(=O)Nc1cnn(C(C)C)c1)CCC C=C(Cl)CC(C(=O)NC(CO)C(=O)OC)NC(=O)CCCCOCC C1(NC(C2ON=C(CC)C2)=O)CN(C(c2csc(S)n2)=O)CCC1C(F)(F)F CC(O)CCCCCC(=O)N1CCC2CN(C(=O)COC3CCCC3)CC2C1 c1(C(=O)NCC2N(c3c(F)cnc(C)n3)CCC2)cccc2c1ccn2C c1(C(=O)NCC(C)(C(C)C)NC(c2cc(C)sc2)=O)ccc(NC2CC2)cc1 CC(C)CC(CNC(=O)CC1SC(=N)NC1=O)NC(c1conc1C(C)(C)C)=O c1(C(N2CCC3(N(C(C4CC(SC)C4)=O)CCC3)C2)=O)ccc2nnn(O)c2c1 N1(C(C)C)CCCC1C(N1CCCC1C(C)NC(c1cnnn1C1CC1)=O)=O N1(C(Cn2cc(-c3ccc(N)c(F)c3)nn2)=O)CCCC2OCCC2C1 c1(SC)cc(NC(c2cnc(CNC(C3CCCN3C(N)=O)=O)nc2)=O)ccn1 N1(C(C(CSC)(C)C)=O)CC(C)(C(=O)N(C)C(C)C)CC1(C)C.C1CC(=O)N1 N1(C(c2n[nH]c(=N)[nH]2)=O)CC2(CC2)CC1CNC(=O)CN1CC2CC2C1 c1(C(C)NC(C2CC2c2cccc(Br)c2)=O)cc(F)c(N)cc1F c1(OC(CC)C(=O)N(C)C)ccccc1CC(n1cc(-c2ccc[nH]2)nn1)C N1(CCC(C(=O)OC)(C)O)CCC2(CC1)OC(=O)NC2=O c1(C(=O)NC2CC(CNC(c3c(N)sc(C)c3C)=O)C2)cn2ncccc2n1 c1(N2CCC(C3N(C(c4cn(CC)nn4)=O)CCC3)C2)cc(C)c(C#N)c(C)n1 C1(OC)CC(CNC(=O)C=C2CCCCC2)(NC(=O)CCN2CCCC2=O)C1 N1(C(c2ccc(OCC)cc2C)C(=O)NC(C)(C)CC)CC2CC(C)OC2C1 O=C1CS(=O)(=O)CC(C(N2CCC(CF)(NC(=O)Cc3nncs3)C2)=O)N1 C(=O)(CS(=O)(=O)c1ccccc1F)N1CC2CC(NC(C3(CC)CC3)=O)C2C1 N1(C(CC)=O)C2CCC1C(CNC(=O)C(c1cccc(C)c1F)O)C2 C1(C(N2CC(NC(CCCC)=O)CC3(C2)CCC3)=O)CSC(c2ccccc2)=N1 C(c1ccc(OCCNC(=O)C(F)=C(C)C)cc1)=CC(=O)OC c1(C(=O)NCC2(NC(CNS(N)(=O)=O)=O)CCOCC2)cc(Cl)ccc1O c1(OC)cccc(C(C)=CC(=O)NC23CCCN(C(=O)CC4CCC4)C2C3)c1 CC1(C)C(O)C(O)C1NC(=O)CONC(C1CCC(=O)N1)=O c1(C(=O)NCCC(C)NC(c2ccc(F)o2)=O)ccc(SC(F)(F)F)nc1 C=CCC(C)(C)CC(=O)NCCC(C)NC(C1CCC(=O)N1)=O CC(F)(F)CCC(=O)NN1CCCC1C(=O)NC12CC=CC(C1)OC2 C12(NC(c3scc(C(N)=O)c3)=O)CCC(CC1NC(c1ccc(F)cc1)=O)C2 c1(C(N(C(C(=O)NCc2ccc(CC)cn2)C)CC)=O)cc(C)c(C)cn1 N1(C(c2nn(C)c(Cl)c2Cl)=O)CCOc2ccc(Cl)cc2C1 C1(C(=O)NC(C#C)C)CCCCN(C(C2CC(C)(C)CCO2)=O)C1 S1(=O)(=O)c2ccc(c(F)c2)NCC2CCCC(C2)N1.C(C)(C)(C)OCCSC C1(n2cc(C=CC)nn2)CC2CCC1(NC(c1cnc(C(F)(F)F)cn1)=O)C2 S(=O)(=O)(c1cccc(Br)c1C)N1CC2CN(S(Cc3c(C)ncs3)(=O)=O)C2C1 C(=O)(CC(C)(C)CC(F)F)N1CCC(CN=c2[nH]nc(C(C)C)o2)(C)C1 C(C(CC(=O)N1CCC(C(C)O)C1)C1CCC1)NC(c1ccn(CCC)n1)=O c1(OC)cccc2c(C(=O)NCC(C(C)C)NC(=O)C(C)C)cnn12 C1(=CC(=O)NC(C(C(C)C)NC(C(C(C)C)OC)=O)C)C2CC3CC(C2)CC1C3 CC1(NC(C2COC(=O)N2)=O)CCCN(C(=O)CC2(O)CCC2)C1 N1(C(C(C2CCOCC2)C)=O)C(C(=O)NCCNC(=O)C2CC2)CCC12CC2 C(CC(CC)C(=O)NCC1(O)CN(C(C2CCC=CCCC2)=O)C1)=CC c1(Nc2c(C(N(S(C)(=O)=O)CCOC)=O)cccc2)c(F)ccc(Br)c1F C1(C(N(C2CN(C(Cc3n[nH]c(=NC)s3)=O)C2)C)=O)CCc2ccccc2O1 C=CC1OCCC1C(=O)N(CC(=O)Nc1ccc(CC)nc1)C1CCC1 Cc1cccc(C)c1C(=O)NC(CC(C)C)c1ncnn1C C1(CC(=O)NCCN(CCCF)C)CCCCN1C(=O)CC1(C)CCC1 N1(C(C2N(C(C3CN(C)C(=O)N3)=O)C3CCC2C3)=O)CCC12CCC(C)CC2 Cc1nc(C)c(CC(N2CCC(N(CCO)C(c3cc[n+]([O-])cc3)=O)C2)=O)s1 Cc1ccc(C(=O)NC(C)CNC(=O)C(F)(F)c2nccs2)cc1N C1(NC(c2c(CC)non2)=O)CCCC12CCN(C(c1cc(Cl)ccn1)=O)CC2 C=CCCCCCCC(=O)N1CCSCC1CCNC(c1cnc(O)n1CC)=O n1(CC)c(C(=O)NCC2(O)CC(C(=O)NC3CC4(CCC4)C3)C2)cnc1O c1(C(=O)NC2(C3N(C(CC(CC)O)=O)CCCC3)CC2)c(Cl)ccc(F)c1C c1(C(C(=O)NC(CC)CNC(C2(C(F)F)CC2)=O)=O)cnn(C)c1 C#Cc1ccc(C(N2C(C(N3CCC(CC4CC4)C3)=O)CCC23CC3)=O)nc1 C1(CC)CN(C(c2cncc(C)n2)=O)CCN1C(c1ccc(C(C)(C)C)nc1)=O N1(C(c2cc(CC)[nH]n2)=O)CCCC(CCO)CC1.C1C(O)CC(=O)ON1 C1(NC(C(C)Cn2ccnc2)=O)CN(C(c2cnnc(O)c2)=O)CC2(CCC2)C1 c1(CC)ccc(CN(C)C)cc1.C12CN(CC1C)C(=O)CNC2=O.C(C)(C)S c1(-c2ccccc2)c[nH]c2ccc(F)cc12.CCN=C(NCCCC1(C#N)CC1)N c1(Cc2cn(CC(CCNC(CCCCC)=O)F)nn2)cc(OC)ncc1Cl CCC(CCCC(=O)N1CCC(N(C)C)C(C)C1)NC(C1CCC(C#N)CC1)=O C#Cc1cnc(C(=O)NC2CC=C(C(=O)N3CCC(O)(CC=C)C3)C2)c(C)c1 N1(C(C(CC)Sc2ccccc2)=O)CC2(CCC(NC(=O)COCCF)CC2)C1 C1(CN(C(c2c(CC)scc2)=O)CC)CN(C(=O)C(C)(COC)OC)CCO1 c1(C(N2CC(C)C(CNC(=O)CCCS(C)(=O)=O)C2)=O)ccsc1S(N)(=O)=O C(=O)(C1=COCCC1)N1C(C(=O)NCCC(C)O)CCC1C C1(C(N2CC(CNC(c3c(CC)occ3)=O)(OC)C2)=O)CC(F)CN1C CCC(O)C(F)(F)C(=O)NC(=O)C(C)Cc1cccc(C(C)(C)C)c1 C1(NC(C(C(C)(C)C)O)=O)CC2CC1CN(C(c1nccn3nccc13)=O)C2 O=C(C1=NOC2COCC12)NC1CCCCC1NC(=O)CCCCn1ccnn1 c1(CNC(c2c(Br)ncc(C)c2)c2nnnn2C2(C)CC2)cc2cnccc2o1 C1(O)(CN(C(C(CC)C)=O)C)CCN(C(c2ccccc2-n2cccn2)=O)CC1 c1(C(N2CC(C)C(CNC(=O)C=C(Cl)Cl)CC2)=O)ccc2nc(O)oc2c1 N1(C(c2c(OCC)cccc2)=O)CCCCC2(CCN(C(=O)C(C)=O)C2)C1 c1(C(=O)NCC(C)N(C(=O)C(C)OC(C)(C)C)CC)cccc(N)c1C(F)F Cc1[nH]nc(C(F)F)c1C(=O)NCC(CO)NC(=O)Cc1cnn(C(C)C)c1 c1(OC)cccc(OC(=O)COc2cccc(C)c2)c1 c1(C(=O)NCC2(OC)CCN(C(=O)CCCC(C)O)C2)ccc2n[nH]cc2c1 C1(CN(C(c2ccc(C)n2C)=O)C)CN(C(c2cnns2)=O)CC12CC2 c1(NC(=O)C(N2CCCC(c3nncs3)C2)=O)ccc2cncn2c1 c1(OC)nc(C(=O)NC23CC(C2)N(C(c2ccnn2CCF)=O)C3)cc(O)n1 C(=O)(N=c1ccn(CCO)[nH]1)C1CC(COC)CN1C(=O)CCCCSC C(=O)(CC(O)CC1CC1)NCC1C(NC(CCc2cn(C)nc2)=O)C1 C(=O)(C1CCc2nccn21)N1C(CCNC(C=CC(=O)N(C)C)=O)COCC1 CC1CCOCC1C(=O)N(C)CC1(O)CN(C(=O)Cn2ccnn2)C1 CCCC(C(=O)OC)C(=O)N(CCCNC(c1cccc(C(C)(C)C)n1)=O)C1CC1 C(=O)(C(C)C(C)S(C)(=O)=O)N(C(CC)CNC(=O)C(CC)N(C)C)C c1(OC)ccc(C=CC(N2CCCN(C(C3CNC(=O)N3)=O)C(C)C2)=O)cc1F CC(C)CCCCCC(=O)N1CC(C(N2CC3CN(C)CC3(C)C2)=O)C2(CC2)C1 C1(C(=O)NC2CCCN(c3nc(C)c(C#N)cc3)C2)CCCC2(C1)CC2(F)F C(C(CC1CC1)C(=O)N1CC(CCN(C)C)C1)NC(CN(C(C(C)C)=O)C)=O c1(NC(CC(C)O)C)ccncc1S(=O)(=O)NCC(C1CCCCC1)(C)C C1(NC(c2cc(Br)co2)=O)C=CCN(C(=O)Cn2cc(CO)nn2)C1 C=CCCCCCCCCC(=O)NC1CS(=O)(=O)CC1NC(C1CC(O)C1)=O c1(C(=O)NCC(C)CNC(C2(C)COCCO2)=O)cnc(O)c(F)c1 c1(C(=O)NCC(CN(C(C(C2CC2)SC)=O)C)C)[nH]c2c(F)cc(F)cc2c1C S(=O)(=O)(c1ccc(NC(=O)Cn2cc(Br)cn2)cc1)NC(CCSC)CCO c1(C(=O)Nc2ncc(F)cn2)ccc(C2CC2)nc1O.CCCC1C2(CC2)N1 Cc1cc2c(C(=O)NCC3(CNC(=O)CC(C)F)CC3(F)F)cccc2o1 CC1=C(C(=O)N(C2CC3CC2N(C(=O)CCC2CCOC2)C3)C)SCCO1 c1(OC)ccccc1CC(=O)N(CCNC(c1cnn(C)c1C1CCC1)=O)C(C)C c1(CS(=O)(=O)Sc2n(C(C)C)cnn2)nn(C)c(N2CCCC2)c1C1CC1 S(=O)(=O)(c1ccc(C(=O)NC(C)CCN(C(=O)C(C)P(C)(C)=O)C)o1)NC N1(C(CCC(C)C)=O)CCCC12CCCN(C(=O)CC1=NNC(=O)C1)C2 CC(C)C(O)CC(=O)N1CCN(C(c2ccc(C(F)F)cn2)=O)C(CCO)C1 Cc1cc2[nH]c(=O)c(C(N3CCN(c4ccc(OCF)cc4)CC3)=O)cn2n1 c1(CSC(C(=O)N(CCOCCN(C(=O)CCOC)C)C)C)cccnc1 CCC(CNC(=O)Cc1n[nH]c(C)n1)(CC)NC(=O)C(F)=C(C)C C1(NC(CN(c2ccc(C)cc2CCC(C)=O)CC)=O)CC2CN(C(C)=O)CC12 C1(C(=O)NCc2c(C)snn2)CC(O)CN1C(=O)CCSc1ccccc1 C1(OC)(CNC(=O)CSc2ccccc2F)CCN(C(=O)C=CI)C1 C(=O)(CC(C)(C)OC)NCC1(OCC)CCCC1.C(=O)(CN(C)C(C)=O)NCC N1(C(C(C)(C)CCCNC(c2ccc(=N)[nH]n2)=O)=O)Cc2cccc(O)c2C1 C(CCCCC(=O)NCC(N1CC=CC1)=O)n1cc(CC(C(C)(C)C)O)nn1 c1(NC(C)=O)sc(Cl)cc1C(=O)NC1CCN(C(C2CCOC2)C)CC1 C(Cn1cccn1)(C(=O)N1OC2CCC1CC2)NC(c1ccc2nccn2c1)=O c1(CC)ccc(C(N2CCC2(C)C2CC2)C(=O)NCc2ccco2)c(F)c1 C1(F)(CNC(Cc2c(CC)cccc2)=O)CCCN(C(c2cnc(C)[nH]2)=O)C1 C1(C(N2CCC(F)(C(=O)OC)C2)=O)CC2CN(C(=O)CCc3cncs3)CC2C1 C(CC(C(C)(C)C)C12CC(C3C(C)C3)(OC1)C2)NC(=O)NCC1CC(C)(F)C1 C12(C(N3CC(C)C(C(=O)NCC(F)C4CCC4)C3)=O)CCC(CC1F)C2 N1(C(COC)=O)CCC(C2CCCN(C(=O)CC(C)CC(C)(C)C)C2)CC1 c1(N(C2CCOCC2)Cc2cccc(C)n2)ccnc2c1ccn2C C12(CNC(c3cc(C(C)C)no3)=O)CCC1CCN2C(=O)Cn1cccnc1=O C1(O)(C(C)NC(c2c(C)noc2C)=O)CCN(C(=O)C(C)C2CC2)CC1 C(=O)(C1CCCc2ccnn21)N(CC(C)NC(c1coc(C(F)(F)F)n1)=O)C c1(C(=O)NCC2C(NC(C3(C)CC=CCO3)=O)C2)cncc(N)n1 N1(C(c2scc(OC)c2)=O)CCC(C(F)CNC(C2CC2C)=O)CC1 Cc1cc(C(=O)NCCCN(C)C(c2ccn(C)n2)=O)[nH]c1C#N c1(C(N2C(CCNC(Cc3c(C)cccc3)=O)COCC2)=O)ccc(F)c(C)c1 c1(C(N(C)CC2(NC(C3CN(C)C3)=O)CC2)=O)ccc(C(N)=O)cc1F c1(C(C)=O)cc(C(=O)N(C2CC(NC(=O)CC3CC4CC4C3)C2)C)c(C)o1 C1(C(N2C(C)CN(C(=O)CCCc3nccs3)CC2)=O)CCn2nnnc2C1 c1(CCC(N2CCC(CNC(C3CC34CC4(F)F)=O)C2)=O)cncc(Br)c1 C1(C(=O)OC)CCCCCCN1C(=O)C(C)(C)C N1(C(C(=O)NCC)=O)CCCC(C(C)NC(C2(COC)CCCO2)=O)C1 c1(C(=O)Nc2ncc(Br)c(C)c2I)cc2c(F)c(F)ccc2s1 CC#CCC(C(=O)N(CC1=CCSC1)C)NC(c1cc(C(N)=O)c[nH]1)=O N1(C(C(COC(C)C)NC(=O)C=NOC)=O)CCN(C)CC1CO O=C1CC(c2ccccc2)N(C(=O)C(O)C2CCC2C(F)(F)F)N1 c1(C(N2CCC(O)(CNC(CC=C=C)=O)C2)=O)cc(C)c(C#N)c(C)c1 C1(CCNC(C2CC=C(C)CC2)=O)CN(C(=O)C#CC(C)(C)C)CCS1(=O)=O c1(C(N2CCN(C(C3CCC3F)=O)CC2)=O)ccc([N+](=O)[O-])c(C(F)(F)F)c1 c1(CNC(c2c(C)cc(C)o2)=O)nc(CNC(=O)C(C)(C)C2CCCO2)cc(O)n1 c1(NC(CCc2cnn(C)n2)=O)ncnc(Cl)c1F.c12ccc([nH]1)C(=O)C2=O O=C(N=c1nc(Cc2cccc(Cl)c2Br)[nH]s1)N1CCCC1 C(=O)(CCCN=[N+]=[N-])Nc1nc2sccc2s1.C12(CC)CN(C1)C2=O N1(C(Cc2scc(C)n2)=O)CCC(CNC(=O)Cc2cn(C(C)C)nn2)(OC)C1 c1(C(=O)NCC(CO)NC(C(C)c2cccs2)=O)cc(Cl)ccc1N CC1CC(C(N2CC=CC(NC(=O)C(C(C)(C)C)C3CCC3)C2)=O)CC(C)O1 Cn1ncc2sc(C(N3CC(NC(=O)C4=COCC4)C(C4CC4)C3)=O)cc12 C(C(=O)N1CCCC1CNC(c1cnc(-c2cnccn2)s1)=O)(C(C)(C)C)SC c1(-c2nc(CC)nn2C2CCCCC2C)cc2ccc(I)cc2[nH]1 C12(C(=O)OCC)CCC(NC(c3cc(Br)ccc3F)=O)(CC1)CC2 c1(N2CCC(c3cc(C)[nH]n3)C2)nc(NCc2scnc2C)c2ncn(C)c2n1 c1(OC)cccnc1CCC(=O)NC1CN(Cc2cccc(CO)c2)CC1O c1(CN(c2nncs2)CCCNC(C(C)(C)OC)=O)cccc(C(F)(F)F)c1 c1(C(=O)NCC2N(C(c3nccc(COC)c3)=O)CC2)cc(SC)ccc1C C1(=O)CCS(=O)(=O)NC2CC(C2)N1C.c1(NC(CC(C)C)=O)cccc(CO)c1 N1(C(c2nc(C(=O)OC)oc2)=O)CC(CNC(c2ccnc(O)c2)=O)C(O)C1 CC(CNC(=O)CCc1cnccn1)CC(=O)NCC1CCCC(CO)C1 C(=O)(CC1=CCCC1)N1CCC(C(C(=O)N(c2cccnn2)CC)F)C1 n1(CC(=O)N(CCNC(=O)C(C)CC=Cc2ccccc2)CC)cccc(N)c1=O C1(CCOC)(NC(c2cn(CCC)nc2)=O)CCN(C(c2cccs2)=O)C1 c1(N2C(c3c(N)non3)CCC2)nc(Cl)nc2cccc(F)c12 N1(C(CCC(C)O)=O)CC2CC1CN(C(c1n[nH]cc1Br)=O)C2 c1(C(N2CC(NC(Cc3c(C)noc3)=O)C(F)CC2)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2cccc(OCC)c2)=O)CC2(C1)CN(C(c1cncc(C)n1)=O)C2 N1(CC)CC(C(N2CC3CC3(NC(C3NC(=O)C4CC34)=O)C2)=O)CC1=O CCC(C)(C)C(O)C(=O)NCC(C(N1CC(CO)CC(C)(C)C1)=O)OC CC1CC(N(C(=O)CCC2(C)CN(C(=O)CP(C)(C)=O)C2)C)CCN1C.CN c1(CC)oc2ccccc2c1C(=O)NC1CC2CN(C(=O)C=C(C)C)CC2C1 c1(C(=O)NC2CCC(CNC(C=CC=CC)=O)C2)cc2ncccc2o1 N1(C(CC2(OC)CCC2)=O)CC2CCC(CNC(C3CCS3(=O)=O)=O)C2C1 c1(CC)nnc2n1CCCC2C(=O)NC1CN(C(c2cn(C)nn2)=O)CC1(C)C C1(CC(=O)NCC(CCCC)NC(=O)C(C)C(C)COC)CCCC(C#N)C1 C(=O)(CCCC(=O)NCCCOCCNC(=O)C(C)C1(O)CCC1)OC N1(CC=Cc2ccc(C)o2)CCN(CC(N)=O)C(=O)C1 N1(C(CC2(COCC)CC2)=O)CCC2(CC2)CC1C(=O)N(C1CCSC1)C c1(C(N2CCC(C)(NC(C(Br)=C(C)C)=O)CC2)=O)cc(Cl)c(F)cc1O CC1(CS(C)(=O)=O)CCN(C(c2ncc(Cc3cccnc3)s2)=O)C1 N1(C(C(CC(C)C)O)=O)CC2CCC1C(CNC(C1C(F)(F)C13CCC3)=O)C2 C1(CCC)CCCN(C(=O)CCC(C)NC(=O)CCSC)C1 C1(CNC(COCCC=C)=O)CC12CCN(C(=O)C=CCOC)CC2 C1(C(=O)NC(C(C)NC(CC2CCN(C(C)C)CC2)=O)CC)CC2(CCCC2)C1 C#Cc1ccc(C(N2CC(NC(c3c(O)cccc3Cl)=O)CC2CO)=O)cc1 CC1(C(N2CC3CCC3(CNC(c3cccnn3)=O)C2)=O)CCCS1(=O)=O N1(C(CCOCC(C)C)=O)CC2CC1CC2NC(c1ccc(Cl)s1)=O Cc1c(Br)ccc(C(=O)N(CC(O)CNC(=O)C(C)C2CC2)C)c1N C1(CC=C)(C(=O)NC2(CO)CC=CC2)CCN(C(=O)C(c2ccnn2C)C)C1 C1(NC(C(CC)OC)=O)(CC)CCCN(C(=O)C(c2cnn(C)c2)OC)C1 c1(CC)ccc(C(=O)NC2(c3cn(CC(=O)OC)nn3)CCCOC2)c(C)n1 N1(C(c2ccc(C)c(CO)c2)C(=O)NCCC2(C)CC2)CCC2(CCCN2C)C1 c1(CC(=O)N(C)CC2CCCN2C(=O)Cc2ccn(C)n2)ccc(O)c(O)c1 N1(C(CS(C)(=O)=O)=O)CC2CC1CC2NC(c1cc(O)n[nH]1)=O C(CC(O)C(=O)NC1CN(C(=O)OC(C)(C)C)C1)OC(c1cn(C(C)C)nc1)=O C1(C(=O)NCCn2c(C)ccn2)CC(C)CN(C(=O)CCC2CCOCC2)C1 CCC(CC(=O)NCC1(CCNC(=O)COc2cc(C)on2)CCCC1)C(C)C n1(COC)nc[nH]c1=NC(=O)N1CC2(CC(N3CCC(O)C(F)C3)C2)C1 C1=C(CN=c2[nH]c3c(c(=NCC4CC5(CCOCC5)CO4)[nH]2)SCC3)COCC1 N1(C(C2C(NC(C(C)CC3CC3)=O)CC=CC2)=O)CCC12CCSCC2 c1(C(=O)OC)ccc(OCCNC(=O)N(C)Cc2ccnn2C2CC2(F)F)cc1 CC1(C(=O)NC2C=CCCC2C(=O)NCC2C3CCCC23)CCC2CC2C1 c1(C(c2nnnn2C)Nc2ccc(C)c(CO)c2C)nc2cc(F)ccc2[nH]1 c1(CCCC(=O)N2CCC(CNC(C3CCCC34CC4)=O)C2)ccc(Cl)cc1 C12(COC)COC(C(N3CCC(N(C(=O)Cc4sc(S)nc4C)C)C3)=O)(C1)C2 C1(C(=O)NC2CN(C(c3nnn(CC)c3C)=O)CC(C)C2)CC2C=CC1CCC2 CCC(C)(C)CC(=O)N(CC(N1CCC(O)(C(N)=O)C1)=O)CC(C)C N1(C(c2cccn2Cc2ccccn2)=O)CCC2CCCC12 c1(C(=O)NC2C(NC(COC)=O)CC2)cc(F)c2cn[nH]c2c1 c1(NC(CNc2cncc(C(=O)OC)c2C)=O)cc2ccccc2cn1 c1(CN2CC(C(=O)Nc3c(C(=O)OCC)scc3)C2)cc([N+](=O)[O-])c(C)cc1Br C1(C2CC2)(CNC(c2cnc(C)nc2C(C)C)=O)CCN(C(=O)CC2CC2)C1 S(=O)(=O)(c1ccc(NC(=O)C(O)CCC(C)C)cn1)NC C(=O)(C1=NOC(C)C1)NN(CCCCCCC)C(c1ccccc1)=O Cc1ncnc(C)c1C(N1CCC(N(C(=O)C(c2ccc(Cl)cc2)C)C)C1)=O c1(C(C(=O)NC(C)(C)C)N(C2CCOC2)C)cc(Cl)cs1 CC(CC(=O)N1CCN(C(=O)COC2CC2)CC1C1CCC1)C(C)(C)C C(C(=O)NC1CC(NC(c2ccnn2C2CCC2)=O)C1)(C(C)(C)C)OC C1(NC(CC(C)C2CC2)=O)CC12CCN(C(c1cccc(N(C)C)c1)=O)CC2 CCCCCC(O)C(=O)N1CC2CCC1CN2C(=O)CC1CC2CC2C1 Nc1nc(Cl)cc(Cl)c1C(=O)NC1COCCN(C(c2ccccc2)=O)C1 N1(C(CCOC)=O)CCOC(CNC(=O)C=CCOC2CCOCC2)C1 c1(C(=O)NCCCN(C2CCCC2)C(C2CCC2(F)F)=O)cc(O)nc(O)c1 c1(C(=O)NC2C(CNC(CN(C)CC)=O)C2)ccc(Cl)c(Br)c1F C(=O)(C1=CCCCO1)NC1(C2N(C(c3ccc(N(C)C)cn3)=O)CCC2)CC1 C1(NC(C(C)CC2CCC2)=O)CCCCN(C(c2ccccc2C(C)(F)F)=O)C1 C1(CNC(c2n(CC)ncc2)=O)COCCN(C(c2ccc(N)cc2OC)=O)C1 N1(C(c2c(CS(C)(=O)=O)cccc2)C2CC2)CCOC2(CCCNC2)C1 C(C(C(=O)N1CCCC1c1cn(CCCCCO)nn1)N(C)C)OCC C(CN=c1nc(N2CCC(SC)C2)c2c([nH]1)CCOC2)NC(COC)=O S(=O)(=O)(c1cc(NCC2(Cc3ccccc3)CCOC2)ccc1Cl)NCC=C N1(c2ccnc(C(=O)OC)n2)CC2(CC2)CC1CNC(C12CC=CC(C1)OC2)=O c1(CNC(=O)CNC(C2(c3cc[nH]n3)CC2)=O)ccc(O)c(F)c1 C(=O)(C1=COCCO1)NCCCC1OCCN(C(C2CCN(C)C2)=O)C1 C1(C(=O)NCC2CC(=O)NCC2)CCN(C(C2CCCCC(=O)N2)=O)CCO1 C(=O)(C(C)(C)CC(F)F)N1CCC(C(C)CC(=O)NC(C)(CO)CO)CC1 c1(C(CN(C(=O)CN2CSCC2=O)CCC)OC)ccccc1 c1(C(C(=O)NC(CN(C(COCCOCC)=O)CC)C)C)c(C)n[nH]c1C c1(C(N2CCC23CCC3)C(=O)NC(CC)(C)C)ccc(F)c2c1CCC2 N1(C(C(N2CCCCC2C2CC2)=O)=O)CCNCC1c1cccc(Br)c1 c1(OC)nc(Cl)ccc1C(=O)N(C1CCCN(C(=O)C(C)(O)COC)C1)C c1(C(=O)NC(CNC(=O)CCC2CNC(=O)N2)C2CC2)cccc(C(F)(F)F)c1 CC1(CCO)CCN1C(C1(CNC(=O)C(C)(C)n2cnnn2)CC1)=O c1(C(N(C)CCNC(C23CCC(F)C2CC3)=O)=O)ccc([N+](=O)[O-])cc1 N1(C(=O)NC2CC(O)C(F)C2)CCCCCCCC1 c1(OC(C)C)cccnc1C(=O)NCC(O)CCNC(c1ocnc1C1CC1)=O C(C(=O)OCC(F)(F)Br)(C(C)C)OCC(C)C.c12ccccc1NC2=O Cc1ncc(C(N2CC(NC(C3CCC34CCC4)=O)CC2CO)=O)c(=N)[nH]1 C(C)(CCCCNC(=O)Cc1cccc(C(C)(C)C)c1)NC(C(C)OCC#C)=O Cc1cc(C(=O)NC2C=CCC2)cc(C)c1OC(F)F.N12CCC1CNC2=O C=C(C)CC(C(=O)N(C)CC1(C)CC1)NC(=O)C1CC1 c1(CCC(=O)NC(CC=C)CNC(C)=O)ccc(S(=O)(=O)CC)cc1 N1(C(C(N2CCCC(O)C2)C)=O)CCC(F)(C(=O)NCc2ccncc2)C1 CN1CCOCC1CNC(=O)C(=O)N(CC1CCCC2CC12)CC1CCCOC1 C1(F)(CNC2CC(N(C)C)C2)COCCN(C(=O)OC(C)(C)C)C1 N1(C(C(C)(C)N(C)C)=O)CCC(C2CC(NC(c3nn(C)c(Cl)c3Cl)=O)C2)C1 Cc1ccc(C)c(NCC(N2CCCCC2C(C)NC(c2ccccn2)=O)=O)c1 C=CC(CC)CC(=O)NC12COC(CNC(C3CCCN3S(C)(=O)=O)=O)(C1)C2 C(=O)(CN=S(C)(C)=O)NCC1N(C(CC2N(C)CCOC2)=O)C1 c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CCOCC1NC(=O)C(F)CC1CC1 C1(CNC(C2C(C(=O)OC)C2(F)F)=O)CC2CCC1N2C(=O)CC1CC(C)(C)C1 c1(C(N2CCC(C3(c4cccc(Br)c4)CCCC3)CC2)=O)cccc(C2CC2)c1 N(C(=NCCCF)NC1CCCSC1)C(Cc1ccc(C)cc1)C Cc1nn(C)c(-c2ccsc2)c1C(=O)NC(C)CC(C)NC(C1CC(O)C1)=O CC(CC(=O)NC1CCC(NC(=O)Cc2c[nH]ccc2=O)C1)C1CCCCC1 N1(CCCCOC)Cc2ccccc2CC1CNC(C1CCS(=O)(=O)N1)=O c1(C(N2C(CCNC(C(C)(C)OCC)=O)CCC2)=O)cc(F)c2[nH]nnc2c1 C#Cc1ccc(C(=O)NCC2CC3CC3N2C(c2ccc(Br)cc2N)=O)nc1 Cc1nn(CC(=O)NCCC(C)(C)CNC(=O)C(C)CC#N)cc1[N+](=O)[O-] c1(C(N2CC(NC(C(C)(C)CC#N)=O)C(C)(C)C2)=O)nccc2cccnc12 C(=O)(C1CCCc2nn(C)cc21)NC1CC2CN(C(c3c(C)nc[nH]3)=O)CC2C1 c1(CC(=O)NC2(C(N3C(C(N(C)C)=O)CC3)=O)CCC2)cc(C2CC2)no1 C(=O)(C#CC(C)(C)C(F)F)N1C(C)C(c2ccccc2)CCC1 C1(CNC(C(CC)CC)=O)CN(C(c2cn(C3COC3)nn2)=O)CCC1(C)C c1(CC)ccsc1C(=O)NC(c1nocc1C(=O)N(CC(F)Cl)C)C C1(CCCCNC(C23CC(C)(C2)C3)=O)CCCN(C(=O)CCn2ccnc2)C1 C1(CC(N2CCC(NC(C3(c4cccs4)CC3)=O)C2)=O)CCCC1(F)F c1(CC)ccsc1C(=O)N(CC(C)O)CCO.C1=CCNC1=O N1(C(c2cc(OC)ns2)=O)CCN(C(c2ccc3cccnn23)=O)CC2(CC2)C1 C1(CC)CN(C(=O)Nc2ccc(NC(C)C)cc2)CCN1C(c1nccn1C)C c1(C(C)NC(=O)CCCCNC(=O)COCCN(C)C)ncc(F)cc1F N1(C(c2ccc(OC)nc2)=O)CCc2cc(NC(C3CC3C3CC3)=O)ccc2C1 N1(C(=O)NCC(c2cccnc2)NC(c2nocc2Cl)=O)CCOCC1 N1(C(CCS(C)(=O)=O)=O)C2CCCC1CC(NC(=O)CCNS(=O)(=O)C(F)(F)F)C2 CC(F)(F)CC(=O)N1CCCCC1C(=O)NCC1CCCOCC1 c1(C(=O)NCc2cc(C)c(F)cc2)cc2cc(O)ccc2nc1C c1(C(N2CCC(Cc3c(C)cccc3)C2)=O)cc(F)cc2ccoc12 C1(=O)CC1(C)C.C(=O)(C(C)CN(C)C)NC(CC)CN.C(C)(C)(C)O C1(NC(C(C)SCCCC)=O)CCN(C(c2scc(C)c2C)=O)C1C c1(CNC(N(C2CCN(c3cc(CC)ncn3)CC2)C)=O)ccc(OC)c(C)c1 c1(CC(N2CC3(CCN(C(C)=O)CC3)C2)=O)c(C)nc2nc(=N)[nH]n2c1C N1(Cc2c(OC)cccc2)CCN(C(=O)Cn2cc(Br)cn2)C2CC12 CC(CCCC(=O)NCC1CCC2CC12)NC(C1CC1F)=O N1(C(Cc2c(C)con2)=O)CC(CNC(=O)Cn2nc(C)oc2=O)OC2(CCC2)C1 c1(CN(C(C(C)OCCC(C)C)=O)CCNC(=O)C=CCO)ccccc1 C1(C2CCCN(C(=O)NC34CCC(C3)C4)C2)(NC(C(CCC)OC)=O)CC1 C1(CC(=O)NC2(C(COC)O)CC2)CC2CN(C(C)=O)CC12.C(=O)(C(C)(C)C)N c1(CC(=O)NCCCCCNC(c2c(SC)csc2)=O)c[nH]c2ccc(Cl)cc12 C1(C(N(C2(C(=O)NCC3(C)CC4CCC3C4)CC2)C)=O)CCC(C2CC2)C1 Cc1cc(C(=O)NCC(F)CNC(=O)CNC(=O)C=Cc2ccco2)ncc1Cl C1(C)(CNC(C2(SCC)CC2)=O)CCCN1C(C1CCOC1C)=O N1(C(C(=O)NC(CC)C)CCc2cccc(Cl)c2)CCc2ccncc2C1 C1(CCCC(=O)NCC2(F)CC(CNC(COCC#C)=O)C2)CCCC(=O)N1 C(CN=c1cccc(S(=O)(=O)NCC(c2ccsc2)O)[nH]1)C1(C)CCCC1 C1(CC=C)(CNC(C2CCN2CC)=O)CN(C(=O)COC2(C)CCC2)C1 c1(C(=O)NC(C2(O)CN(C(C3(C#N)CCC3)=O)C2)C)[nH]nc([N+](=O)[O-])c1Cl N1(C(CCCC2(C)N=N2)=O)CCC(O)C(NC(=O)CCC2CCC2)C1 C1(CC(=O)NCC(C)N(C)C(c2cc3[nH]ccc3s2)=O)CC2(CCC2)CO1 c1(NC(C(C)(C)CF)=O)cnc2c(c1)C(=O)NCC2 n1(CC(=O)NCC2N(C(CCCOC3CCCC(C)C3)=O)CC2)ccc([N+](=O)[O-])n1 N1(C(C(n2cc(C3(c4ccccc4)CCC3)nn2)C)=O)CCCC2(C=CCO2)C1 Cc1nnc2n1C(C(=O)NCCCNC(C1(c3ccccc3)CC=CC1)=O)CC2 C(=O)(C1CCc2c[nH]nc21)N1CCN(C(=O)Cn2cncn2)CC1C1CC1 C12CC(F)CN1C(=O)c1ccc(o1)NC2.Cc1nc(CNC(CC(C)C)=O)cs1 N1(C(c2cscc2C2CC2)=O)CCC(CO)(CNC(C2(C(F)F)CCCO2)=O)C1 c1(N(C)C)nc(Cl)c(CC#N)s1.C12CCCC1CCNC(=O)N2.C(C)(C)(C)OC(=O)N c1(OC)sc(C(=O)NC2(CNC(c3ncccc3N)=O)CCC2)cc1Br C1(NC(C(CC#C)NC(=O)CC2CCC(=O)CC2)=O)CCC12CCCC2 c1(CCC(=O)N(C2CCN(C(COC)=O)C2)C)c(Cl)cncc1Cl C(CC(C)C)(C(=O)NCC1CCCCC1C(N1CC(F)CC1CO)=O)OC c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(CC(C)C)(C)C)cnc2n1CCC2 C1(Cc2c(C(=O)OCC)[nH]cc2)CCC(n2cc(C(C)(C)C)nn2)CC1 C1(C(C)NC(C(=Cc2ccco2)C)=O)CCCN(C(c2ccoc2Cl)=O)C1 N1(C(C2CCN(C)C2=O)=O)CCN(C(=O)CCCNC(N)=O)CC1CC(F)(F)F CCCCC(C(=O)N1CC(F)(CNC(C2CCCS2)=O)C1)C(C)C N1(C(C(C)OCCOC)=O)CCC(C(C)C(=O)NCC2(CF)CC2)CC1 C12(CCCC1)C(=O)N2.C1(NC(CN(CCOC)C)=O)CCC1COC Cc1cn2cc(C(=O)NCC3CN(C(=O)Cc4csnn4)CC(C)(C)O3)sc2n1 C(=O)(CN=c1cc[nH]cc1)NCc1nccc(C(N2CCOCC(C)C2)=O)c1 CC1=CCCN(C(=NCCF)NCC2CC(C)(C)C2)C1 N1(C(CC2N(CC)C(=O)CC2)=O)CCC2(C1)CN(C(=O)Cc1cn(C)cn1)C2 N1(C(Cc2c(C)noc2)=O)CCCC2(CCCN(Cc3cc(F)ccc3F)C2)C1 C12(C(=O)NCC3(NC(Cc4cc(COC)on4)=O)CCC3)CC(CC(C)O1)C2 C(C#CCN=c1nc(-c2ccc(OC)cc2)o[nH]1)N(c1ccc(Br)cc1)C c1(CC)nn(C)c(CC)c1C(=O)NCC1(O)CN(C(c2ccn(O)c(=O)c2)=O)C1 N1(C(C2(C)C(CC)CCC2)=O)CCC(CO)(CNC(c2cncc(Cl)n2)=O)CC1 C1(C(=O)NC(CC(=O)OC)(C)C)CN(C(=O)C(C2CCCCC2)=O)CC1(F)F C1(C)(C(N(C2CCN(C(C(C)OCC#C)=O)CC2)CC)=O)COC(C)(C)CO1 N1(C(c2c(NC(=O)Nc3ccccc3)cccc2)=O)CC2C(C1)C2(F)F Cc1ncsc1CNCCOC(C)C.c1(SC)cc(OC)ns1 C=CCC(CNC(=O)CCCCCNC(=O)C(C)CC1CC1)CC(C)C c1(C(N2C(CN(C(C3CCCOC3)=O)C3CC3)CC2)=O)cccc(OC(F)F)c1 N1(C(c2cc(OC)no2)=O)CC2CCC1C1CN(C(c3ccccc3O)=O)CC21 c1(C(=O)NCC(CNC(=O)CCCNC(N)=O)OC)nccc2ncccc12 C1(CC(C)SC2CCCC3CC23)CCN(C(C2(c3ccnn3C)CC2)=O)CC1 N1(C(C2C(NC(CC(C(=C)C)OCC)=O)CCC2)=O)CCC12CCOCC2 N1(C(C(C)N(C)C)=O)CCOC2(CCN(C(=O)Cc3ccoc3)C2)C1 N1(C(COCCCCC)=O)CC(O)(C(C)NC(c2ncnn2C)=O)C1 CN1CCC(C(=O)NCCc2cccs2)(NC(c2ccc(CO)o2)=O)C1 N1(Cc2sc(C(=O)OC)c(C)n2)CC2CCC1CN(C(c1cncs1)=O)C2 C#CCC(C)(C)C(=O)NCC(C1CC1)N(C)C(c1cc2sccc2s1)=O N1(C(c2c(CC)nco2)=O)CC(N(C)C(c2cc(OC)no2)=O)C(O)C1 c1(C(N2CC3C(CNC(C(C(CC)O)C)=O)C3C2)=O)c(F)ccc(O)c1O c1(CC)ccnc(C(=O)NC(CC2CC2)CC(=O)NCC2CC(F)(F)C2)c1 C#CC1(C(=O)N(CC(CC)NC(=O)CCCNC(c2ccco2)=O)C)CCCC1 C(=O)(C1Cc2ccccc21)N1CC=C(CNC(c2c(C(C)C)occ2)=O)CC1 Cc1nn(CC(=O)NCCNC(=O)CN(C2CCC2)C)c(=O)o1 N1(C(C2CCC(=O)NC2)=O)CC2(CCC2)CC1C(=O)NCCC(Cl)Cl C1(NC(=O)C=CCN2CCCC2)CC(F)CN(C(C2Cc3cscc3C2)=O)C1 Cc1cc(Cl)c(C(=O)NC2(C)CCN(C(c3ncccc3F)=O)CC2)cc1C C1(CNC(C(C2CCCO2)SC)=O)CCN(C(=O)COCCN(C)C)C12CC2 C1(CC)C(C(=O)NCC(=O)NCC2CC2)CCN1C(c1ccncc1Cl)=O N1(C(C(C2CC2)OCC)=O)CCN(C(c2coc(C(C)(C)C)n2)=O)CC12CCC2 CC1=NOC(C(N2CCC2CNC(=O)CCc2nc(O)n[nH]2)=O)C1C C(C(C(=O)N1CC=CC1CF)NC(c1cnc(C(C)C)o1)=O)OCC C1(NC(COCC(=O)NC)=O)COCCC1NC(=O)C(F)CC1CCC1 C1(CNC(CC(C=C)C)=O)CN(C(=O)C(C)C)C2COCC2O1 CCC(C)(C(=O)N(C1(CC(=O)N(CC(C)C#N)C)CC1)C)OC CCCCC(O)CC(=O)N(CCNC(c1ccncc1OC)=O)CC C1(CNC(c2cc(CNC(C3C(C)CCO3)=O)sc2)=O)CCC(=O)NC1 S(=O)(=O)(c1cccc(Cl)c1Cl)NCC1OCCN(c2c(C)cnc(SC)n2)C1 c1(OC)nc(Cl)ccc1C(=O)N(C1CCCN(C(=O)CCN2CCC2)CC1)C Nc1cccc(Cl)c1C(N1CCC1CNC(=O)CC1=CCCC1)=O CCC(C(=O)N1CC2CC1C2NC(c1ccc(Cl)cc1C)=O)C(C)C N1(C(CN(CC)CC)=O)CC2C3CCC(C(NC(=O)C(O)CCC(C)C)C3)C2C1 Cc1cccnc1C=CC(=O)NCC1C(C)CCCN1C(c1coc(O)n1)=O N1(C(C(C)Cc2cnc[nH]2)=O)CC(C)(CNC(C2(CO)CC2)=O)CC1(C)C CC(C)(C)C(O)C(=O)N1CC(O)C(O)C1CNC(=O)C(F)=C1CCCC1 C1(N(C(c2c(C)snn2)=O)C)CCC2CN(C(C3CC(O)C3)=O)CC12 C(=O)(C(CCN(CC(CCCC)CC)C)C(C)(C)C)OC(C)=O C=CC(CC)CC(=O)NC1CC(C(C)(C)NC(C2CCOC(C(F)(F)F)C2)=O)C1 CC1(C)Cc2cccc(C(=O)NCC(F)CNC(C3(C)CC3(F)F)=O)c2C1 C1(NC(CCc2ccc(C(N)=O)[nH]2)=O)CCCN(C(C2C=CCC2)=O)C1 C1(NC(C2(COC)CCC2)=O)CCN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC(O)C1 C(=O)(C(F)CC1CN(C(=O)CC2CCC2)C1)NCCCN(C)C N1(C(C(N2C(CN(C(C)=O)C)CCC2)=O)C)CCCCCCC1=O C1(NC(C2(C(C)NC(C3(CN(C)C)CC3)=O)CC2)=O)CCN(C(C)CO)CC1 N12CCCN(CCC1)C(=O)C21CC1.c1(OCC)ccc(OCC)cc1.C(=O)(OC)NC c1(C(C)C)ccc(NCC(N2CC(CNC(=O)Cc3ccco3)C(C)C2)=O)cc1 c1ccc(Br)c(F)c1F.CN1CC(C(=O)OC2CCN(C(=O)NCN)CC2)CC1=O N1(C(C(=O)Nc2cc(OC)c(OCCC)c(Cl)c2)=O)CCCC2(CCSCC2)C1 c1(C(=O)NCCC(C)NC(c2conc2C2(C)COC2)=O)ccc(CO)cn1 C1(NC(CCn2c(C)ncc2)=O)CC2(C1)CC2C(=O)N(CCCO)C1CCC1 N#Cc1cc(C(N2CCC(NC(=O)CCCC(F)(F)F)CC2)=O)cc2[nH]ccc12 C1(C(N2CCCC(CCNC(C3CC3C(C)C)=O)C2)=O)(CC)CCOCC1 C1(CNC(C2ON=C(CC)C2)=O)COCCN(C(=O)CCc2cncc(O)c2)C1 c1(CN2C3C(C(N4CCC(C(=O)OC)C4)=O)C(C3)C2)cc(Cl)ncc1Br N1(C(=O)CC2C=CCC2)CC(O)(C2CCN(C(=O)Cc3ccsc3)CC2)C1 Cc1onc(Cl)c1C(=O)NC(C)CCCNC(c1ccn(-c2ccccc2)n1)=O C1(OC)CC2(C(=O)NC3CC3NC(=O)C(c3cncn3C)OC)CC12 Cc1cccc(C(=O)NCCCCC2CN(C(C3CCCC34CC4)=O)C2)c1N CC(C)C(C(=O)NC1CC1NC(C12OCC(NC(=O)C=COC)C(C1)C2)=O)C(C)C C1(C)(CNC(C(CC(C)C)C)=O)CC(F)(F)CN1C(c1ccc(C(N)=O)s1)=O C1(NC(c2c(C)nncc2)=O)CCC2(CCCN(C(c3ccc(Cl)cn3)=O)C2)C1 O=C(C#CC1CCCO1)NCC1CCN1C(c1ccc(Cc2ccccc2)[nH]1)=O CC(F)(F)C(C)(C)C(=O)NC1CCCC1CNC(c1c(F)ccc(C#N)c1F)=O N1(CCNC(C(CC)O)=O)CCC(NC(=O)CCC2(C#N)CCC2)CC1 c1(C(C)C(=O)NC2CCN(C(=O)CSC(F)F)CC2)cc(F)cc(F)c1 C12(C(=O)NCCCC(=O)NC3CCCC(CC)C3)CCC(n3cccn3)(CC1)C2 c1(C(=O)NC(CCCNC(C2N(CCC)C(=O)CC2)=O)(C)C)ccc(C)cc1C C#CC(CNC(=O)C(C1CCCO1)NC(=O)CC1CCN(C)CC1)C(C)C c1(OC)sccc1C(=O)NC1CCCC1NC(=O)CCN(S(C)(=O)=O)C c1(NC(C2CN(C(=O)CSC(=N)N)CCO2)C)c(F)cccc1[N+](=O)[O-] c1(CNCC2C(F)CCN(C(c3ccc(F)cc3O)=O)C2)cc(O)c(F)c(F)c1 C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(NC(c2cc(C)c(=O)n(C)c2)=O)CC1 CCC(CC)C(C(=O)NCCC#N)N1CCOC(C)(C(C)(C)C)C1 C(C(=O)OCC1CC1C(=O)OC)=CCC C1(NC(C2CCC(NC(c3n(C)nc(O)c3)=O)CC2)=O)CCCC(O)CC1 Cc1cc(Cl)c(C(=O)NC2(CF)CCN(C(C3CCC4(CCC4)C3)=O)C2)cc1F CCC(Cc1cn(Cc2nnc(C3CCCC3)o2)nn1)C(=O)O Cc1ncccc1C(=O)NCCC1CCN(C=O)C1.C1(C)CCCSC1 c1(C(=O)NC2CCN(C(c3n[nH]c(C)c3O)=O)C23CC3)c[nH]c2cc(Cl)ccc12 N1(C(CCC(C)N(C)C)=O)CCC(NC(C2(CF)CCC2)=O)C(C)(C)C1 c1(C(=O)NCCNCCCCn2cccn2)ccc(OCC(=O)NC2CC2F)cc1 c1(CCCC)nc(C)c(C(N2CC3C(CNC(c4nccn4C)=O)C3C2)=O)s1 c1(C(=O)NC2CN(C(C(C(C)C)C3(C)CC3)=O)C2)cc2n(n1)CC(C)NC2=O c1(C(=O)NCC(CNC(C(CC)CC)=O)(C)O)ccnc2cc(F)cnc12 C=CCCCC(C1CC1)NC(c1coc(CNC(=O)CC2(N(C)C)CC2)n1)=O C1(N(C(=O)C(F)n2cccn2)C)CC2CCC(C1)N2C(c1cnc[nH]1)=O Cc1ccc(F)cc1C(N1CCCC(C(C)C(=O)NC2C(O)CC2O)C1)=O CN1CC(NC(=O)Nc2ccsc2)C(F)(F)C1 C1(NC(C(CC=CC)NC(C2CN(C)CCO2)=O)=O)CCCCC1(C)C C1(NC(C2(C(C)C)CCCO2)=O)CCC(C#N)CC1.Cc1coc2c1C(=O)NC2 N1(C(C2OCCN(C)C2=O)=O)CC(NC(C2CCC(=O)N2)=O)CC(C)(C)C1 N1(c2nnc(C(C)C)o2)CCC(C)C(NC(=O)CCc2cn(C)nn2)C1C CCCCC(O)C(C)C(=O)NC(CO)C(=O)NCCCCCC(C)C C(=O)(CCS(C)(=O)=O)NCC1C(NC(CCc2cccc(OC)c2)=O)C1 C12(NC(c3cc(OC)no3)=O)CCCC1CN(C(=O)C1=COCCC1)C2 S(=O)(=O)(c1ccc(NCC2CSCCO2)c(F)c1)NC(CC)CC1CCCCC1 C1(NC(COCCN2CC=C(C)CC2)=O)CN(C(=O)NC(C)(C)C)CC(C)O1 c1(CC(=O)NCCNC(=O)CC2=CCCCC2)ccc(F)cc1[N+](=O)[O-] CC1(C)C(NC(N2CCCC(C)(C(=O)NC3CC3)C2)=O)CC1(F)F CCC(C)C(CC(=O)NCc1cn[nH]c1)NC(c1cn(C)ccc1=O)=O C(CN=c1[nH]c2c(c(=NCC3CCCCO3)[nH]1)CCCC2)c1cc(C)c(F)cc1 CC(C)(C)C(C#N)C(=O)N1CCC(CCC(=O)NC(c2ccsc2)(C)C)C1 S(=O)(=O)(c1cnccc1N(C)Cc1ccco1)NCC(C(C)C)OC c1(OC)cc(C(=O)Nc2ccc(-n3cncn3)c(C)c2)c(N)c(Br)c1 c1(C(=O)NC2C(NC(C(CC)Nc3ccccc3)=O)C2)cc(C)c(C)cc1C N1(C(c2ccnc(C)c2O)=O)CCC(C2(NC(=O)C(C)CC(C)C)CC2)C1 c1(C(=O)NC(CC)CCC(=O)NC2CC3C(CO)C3C2)ccc2c(c1)OCO2 N1(C(CCc2ccc(C)s2)=O)CCC2CN(C(=O)C=CCN(C)C)CCC2C1 CCC(C)CC(C(=O)N(C)Cc1scnc1C)NC(=O)CCCC1CC1 c1(CNC(CCC2(NC(C3C(C(N)=O)C3)=O)CCCC2)=O)cc(F)ccc1F c1(SCC2C(CCOC)CC2)ncnc2c1cnn2-c1ccccn1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(F)c(Cl)c2)C)cccc2c1OCC2 c1(C(=O)NC(C(C)NC(c2c(C)ccc(F)c2)=O)C)c(F)ccc2ccncc12 Cc1cc2cccc(CNC(=O)NC3C4Cc5ccc(Cl)cc5C34)c2o1 S(=O)(=O)(c1cc(C)cnc1NC(C)CSC)N1CC(CCC)OCC1 c1(C(N2CC3CN(C(c4c(Br)cc(C)s4)=O)C3CC2)=O)cc2cc(F)ccc2o1 CCCC(CCC)CC(=O)N1CCC(O)C(NC(c2cc(COC)no2)=O)C1 C1(CNC(c2nc(OC)oc2)=O)COCCN(C(C2CCCC(C)C2)=O)C1 S(=O)(=O)(c1ccc(C#N)c(NC2COC(C)(C)C2)c1)N1CC(CC)N(C)CC1 C1(OC)CC2(C(=O)NCC3(C(C)N)CC3)CCCC12.c1(CC(=O)NC)nccn1C N1(C(CC(C)=C(C)C)=O)CCCCC(CN(C(=O)CCCCC)C2CC2)C1 c1(C(N2CC(F)CC(NC(C(C)=C3CC3)=O)C2)=O)cccc(C2=CCOCC2)c1 C(=O)(C(C)S(C)(=O)=O)NC(CC=CC)C(=O)N1C2CCC1CC2.C(C)(=O)OC C1(C(N(C2CCC2(C)C)C)=O)CCCC1CNC(c1cscc1Cl)=O c1(C(=O)N(C(C2(CC3(CC(=O)OC)CC3)CCSC2)=O)C2CC2)ccnc(O)c1 C12(C(N(C(CC)CC)C3CC3)=O)CC(C)(CN1C(c1ccc(Cl)cn1)=O)C2 CC1(CNC(C2CC(=C3CC3)C2)=O)CCCN1C(=O)CC1(C2CC2)CC1 C1(C2CC2)(C(=O)NC(CC#C)C(=O)OC)CN(C(=O)COCc2ccncc2)C1 N1(C(c2c(C)c(N)cnc2)=O)CCC(NC(=O)CC2C(C)(C)C2(C)C)C(C)(C)C1 N1(C(C(n2ccc(C)n2)C)=O)CCC2(CCN(C(c3conc3C)=O)CC2)C1 CC1c2cc(C(=O)Nc3ccc(CN=[N+]=[N-])cc3)ccc2OC1C c1(C(=O)NC(C(=O)OC)CC2CCCCN2)cccc(C2CC2)n1 S(=O)(=O)(c1cccc(Cl)c1)CN(C(c1ccc(Br)cc1)CC(C)C)CC1CCCO1 N1(C(COCCCC)=O)CCCC(C)(NC(=O)CC(C)(C)C#N)C1 Cc1ccc(C=CC(=O)NCC(C)N(C)C(C2(C)CCCS2(=O)=O)=O)nc1 C1(CN)CC(O)CN1C(=O)N(C(=O)Oc1cn(CC(C)C)cn1)CC1CCCC1 Cc1c(NCC2CCC3(CC3)C2)ncnc1N1CCC(OCc2ccccc2)C1 C#CCCCCC(=O)NCC1CCCN(C(C2CC3(CC3)CO2)=O)CC1 c1(C(=O)NCCCCCNC(C23CCC(OC)C2CC3)=O)c(N)ccc(C)c1F CC(CC(=O)NCC1(F)CCCN(C(c2cc(O)cc(Cl)c2)=O)C1)CC(C)(C)C C1(NC(c2ccc(CC)[nH]2)=O)CCCN(C(=O)C(C(=O)OC)OC)C1 Cc1nc2c(s1)CCCC2C(=O)N1CCC(C)(NC(c2cnn(C)c2C)=O)C1 C(=O)(CC(C)N(C)C(c1cc(C)on1)=O)NC(c1nccn1C)CC N1(C(C(C)SCC)=O)CC(C)CN(C(c2[nH]c(O)nc2C)=O)CC1C c1(C(N2C3CC(CNC(C4N(CC)CCC4)=O)(OC3)C2)=O)ccc2cc[nH]c2n1 N1(C(C(C2CCCC2)OCC)=O)CCSCC1CCNC(=O)COC1CC=CC1 C(CCCC(=O)N1CCC(c2nnc(Br)n2C)CC1)NC(C)=O C1(NC(CCC(CC)C)=O)CC2CCC1CC2NC(c1c(C(F)F)cccc1N)=O N1(C(C(C)(C)OCC)=O)CCC2(CCC(NC(c3ccc(C)n3C)=O)C2)CC1 C(=O)(C#CC1CCC1)N1CC(CNC(CCCc2ccc(CC)cc2)=O)C(C)C1 N1(C(C(CC)=CC)=O)CC2CCC2(NC(c2cc(C#N)c[nH]2)=O)C1 c1(NC(C2N(C(c3c(C)cc(N)cn3)=O)CC(=O)NC2)=O)cnn2c1OCCC2 C#CCCCCC(=O)N1CC(F)CC1CN(C)C(C1OCCOC1C)=O c1(C(=O)NC(c2ccc(CNC(c3n[nH]cc3N)=O)cc2)C)c(F)cccc1F C=CCCC(C)C(C)N1CCC(c2cccc(C(=O)OCCCN(C)C)c2)CC1 c1(C(N2CC(c3cn(Cc4c(OC)con4)nn3)(C)C2)=O)cccc2c[nH]nc12 N1(C(C2N(C(C(C)(C)OC)=O)CC(=O)NC2)=O)CC(C)(C)OC(C)(C)C1 C1(C)(CC)C=C(C(=O)NCC2(COC)CCN(C(C3(C)COC(=O)C3)=O)CC2)C1 C(=O)(C1OC(C)Cc2ccccc21)NCc1c(C)cccc1Br C1(CNC(c2nnnn2CC(F)F)C(C2CCCC2)OC)(CCl)CCOCC1 N1(C(C(N)=O)=O)CC23CCCCC2(C1)CN(C(c1cc(Cl)cc(Cl)c1F)=O)C3 C1(C#N)(C(=O)NC2C(NC(CSCCN(C)C)=O)CCCC2)CC12CCCC2 C1(OCC(C)C)CCN(C(N2CC(C)(CCO)C2)=O)C1 C1(C(N2CCCC(CC(=O)NC(c3ncccn3)CC)C2)=O)CC2(C1)CC(O)C2 C1(OC(F)F)CCCC(NC(c2ccc(CBr)cc2)=O)C1.C=O C1(C(C)NC(=O)CNS(=O)(=O)C2CC2)CCCC(C)(C)O1.N12CCOC(C1)C2=O c1(CC)cc(Br)c(C(C(=O)Nc2ccccc2)N(CC(Cl)Cl)C)s1 N1(C(CC=CCC)=O)CCC(C(N2CC(C(C)C)CCC2C)=O)(CC)CC1 c1(OCC(=O)NC2CN(C(c3ccccn3)=O)C2)ccc2c(C(=O)OC)csc2c1 C=C(Cl)C(C)(C)C(=O)NC1CN(C(C2(F)CC2c2ccccc2)=O)CC1C C1(CNC(c2n(CCCC)ncc2)=O)CN(C(c2ccnc(O)c2)=O)C(C)(C)C1 c1(C(=O)NC(CNC(C(C=C)O)=O)C)cc(Br)c(OC)cc1N c1(C(=O)NCC2CC(F)CN2C(C2CC23CCC3)=O)nccn2nccc12 N1(C(COCC(C)C)=O)CCC2CN(C(=O)Cn3nnnc3C(C)(C)C)CC2C1 c1(C(N(CCC(C(C)(C)C)NC(=O)CCC(N)=O)C)=O)cccc(N=[N+]=[N-])c1 N1(C(COCCOC)=O)CC(OC)CC(C(=O)NC(C)CN2CCCC2=O)C1 c1(C(N2CCC(NC(Cc3ncc(C)s3)=O)CC2C)=O)occ2c1CCOC2 CC(CCC(=O)NOCC(O)CO)CCC(=O)NOC1CC(c2ccccc2)(c2ccccc2)C1.C(C)C c1(C(N2CCC(COC)(CNC(=O)C(O)C(F)F)C2)=O)cc(F)ccc1NC C#Cc1ccc(C(N2CC(NC(=O)Cc3ccc(C)cc3Br)CCC2C)=O)cc1 c1(C(=O)NC(C)(C)CCC2CCCN2C(C2COC(=O)C2)=O)ccn(C)c(=O)c1 N1(C(CCOC)=O)CCCC(C(=O)NC2CC2C(N2CCN(C(N)=O)CC2)=O)C1 O=C1NCc2c1ccnc2C(=O)NCC1CCCN1C(C1CC(=O)C12CCC2)=O C=C(Cl)CC(C(=O)N1CC(C#N)C1)NC(=O)CCC(=O)NCC C#Cc1ccc(F)c(C(=O)NCC(CC(F)(F)F)NC(C2CC(C(F)F)C2)=O)c1 C1(CNC(C2(CN)CC2)=O)COCCC1(F)F.c12cn(nn1)C1CN(C1)C2=O CCCCCC(CNCc1ncc(C)s1)N1CCC(C(=O)NC)C1 C(c1cccc(F)c1Cl)=CC(N1C2C(NC(CS(CC)=O)=O)C(C2)C1C)=O c1(C(N(CC(=O)N(C2CC(C#N)C2)CCCC)C)=O)cnc(O)c(C)c1 C(=O)(CCCCNCC1CCCC(SC)C1)OC N1(CC(N2CCCC(C(=O)NC)C2)=O)CCCC(C)(O)C1 C1(NC(CSC)=O)CC2CCC1CN(C(c1ccnc(N3CCOCC3)n1)=O)C2 C1(O)(CC(=O)N(C)CCN(C(=O)C(c2ncc(Cl)n2C)(F)F)C)CCCN(C)C1 c1(-c2c(C(=O)NCCN3CC4CC4C3)c[nH]n2)cccc(Br)c1.C12CCN1C2=O c1(C(=O)NC(C2CCCCN2C(c2cnn[nH]2)=O)C)ccc(F)c(CCN(C)C)c1 Cc1cc(CC(=O)NCC2CC(F)(CNC(=O)C(C3CCCCC3)O)C2)no1 N1(C(C2(CC)CC2(F)F)=O)CC2(C1)CN(C(c1cccnc1C1CC1)=O)CCO2 c1(C(C2CCCCC2)C(=O)NCC(C)NC(CCOC)=O)ccccc1[N+](=O)[O-].N c1(CC)nncn1NC(=O)CC12CCCC1C2.C1(=O)C(F)CC(=O)NC1=O.OCC O=C(C1=C(Cl)CCCC1)NC1CC(O)CN(C(=O)C(c2cc(F)cc(F)c2)O)C1 c1(OC)ccc(Cl)cc1C(=O)NC(C1(O)CN(C(c2cc(O)nc(O)n2)=O)C1)C C(=O)(C1=CC2CCC=CCCC12)NC(C)CCN(C)C(c1ncccn1)=O CCC(CC(C)C)C(=O)NCc1nc(C(=O)NC2CSC2)c(C)o1 C1(NC(C(CCCC)O)=O)CC2(CCCN(C(C3CCS(=O)(=O)C3(C)C)=O)C2)C1 c1(C(=O)NC2C(F)CCN(C(CC3C(=O)NC(=O)N3)=O)C2)ccc2nc[nH]c2c1 c1(C(=O)NC2CCCN(C(CCc3n(C)ccc3)=O)C2)scc2c1OCCO2 CC1CN(C(=O)CCC2CC2(C)C)CCC1NC(C1CCC(N(C)C)CC1)=O N1(C(C(C(C)C)(C)C)=O)CC2(NC(c3cccc(O)c3Cl)=O)CCCC2(F)C1 c1(CNC2CC(S(N)(=O)=O)CC2)cc2cc(Cl)c(Cl)cc2[nH]1 c1(C(=O)NCC(C(C)(C)C)NC(=O)CCF)cc(N)cc2c1OCCO2 C(CNC(=NCc1ccccc1)NCC1CN(CC)C(=O)O1)(C(F)(F)F)OCC c1(CCC)cc(C(=O)NC2CCCC2NC(=O)CCn2ccnc2)cc(O)n1 N1(C(Cn2c(N3CCC(OC)CC3)nnn2)=O)CC(CN=c2nc[nH]s2)C(C)(C)C1 c1(NCC(N2CCN(C(C=CSC)=O)C3C2C3)=O)ccccc1[N+](=O)[O-] C1(NC(Cc2onc(C)n2)=O)CC(C)CN(C(C2CC(=O)NC(=O)N2)=O)C1 C1(CC=C)(NC(C2SCCCS2)=O)CCN(C(c2csc(C#N)c2)=O)C1 c1(NC(=O)Cc2nc(NC(c3ccccc3F)=O)cs2)cccc(Br)c1F N1(C(Cc2c(C)noc2C)=O)CC2COCC2(C(=O)NCC2CC23CC3(F)F)C1 C12CCOCC1(CC)NCC2O.C1(CC)CC(CO)(CC2(C)OC2)C1 CC(C)C(C(=O)NC(C1CCCN1C(c1cc[nH]n1)=O)(C)C)n1ccnc1 c1(C(N(C2COCC2N)CC)=O)nc2ccc(O)cc2s1 C1(CC)CCCCN1C(=O)COc1cccc(C(=O)NC(C)C2CC2)c1 C1(N(C(CCSCC(C)C)=O)C)CCCC(NC(c2cc(CO)[nH]n2)=O)C1 N#Cc1sc(=NC2CC(C(=O)NCc3nc4ccccc4[nH]3)C2)[nH]c1Cl C1(c2cn(CCC=C=C)nn2)C2CCCC1N(C(c1cccc(F)n1)=O)C2 N1(C(C=Cc2c(C)ncs2)=O)C2CCC1CC(CNC(=O)CCc1nc[nH]n1)C2 C(C)(C)(CC(=O)NC1CC(C(N)=O)C1)NC(C(C1CCCCC1)C)=O O=C(C#CC1CCCCC1)NC1(CNC(=O)CC2CCOC2)CCC(F)(F)CC1 c1(C(N2CCC(n3ccnc3)C2)C(=O)NCCCC)cc(Cl)c2c(c1)OCCO2 c1(OC(C)C)ccc(NC(=O)NC(c2ccc(Cl)cc2)CC2CC2)cc1 C12(F)CCCN(C1)C(=O)C=CC(C)(C)OC2=O.C1(C(=O)OC)CCCN1C(C)=O C1(NC(Cc2nc(C)oc2)=O)CN(C(c2ccc(C)n2C)=O)CC1C1CC1 c1(OC)cc(C(N2CCCC2C(C)NC(=O)C(n2nc(C)cc2C)C)=O)ncn1 N1(C(c2ccc(CCC)[nH]2)=O)CC2CCN(C(c3cc(C(N)=O)co3)=O)CC2C1 c1(C(=O)NC(C)C=CC(=O)NCC(F)(F)CO)ncncc1Cl c12ccc(O)c(c1)CC1CCCN1C2=O.n1(CCOC)cc(CCC2CC2)nn1 c1(CC)ccc(C(=O)NCCOC2CCN(C(=O)C=CCO)C2)cc1 CCC1=NOC(NC(C2CCC(NC(C3(CC)CCCC3)=O)CC2)=O)C1.C1(CC2CC2)CC1 C(=O)(C1=C(C#N)CCC1)N1CC(C)(CCC(=O)N2CC(N3CCC3)C2)C1 C1(C)(NC(CC2CCCC(C)C2)=O)CCN(C(c2cc(C3CC3)ccn2)=O)CC1 c1(CC)cccc(C(=O)NCC2CCN2C(=O)CN2CCCCCC2=O)c1F C#CCCC(C(=O)NC1CCN(CCC)CC1)NC(c1ccc(C)c(O)c1)=O C1(OC)CC(NC(C2CC3CCC(C2)O3)=O)CN(C(c2n[nH]c3c2COC3)=O)C1 c1(C(=O)NCCC2(NC(CC(CC=C)(C)C)=O)CC2)cc2n(n1)CCNS2(=O)=O C1(CNC(C2CSC2)=O)CN(C(=O)C2=COCCC2)CCC1C(F)(F)F C(C1=CCN(C(C2CC(C#N)C2)=O)CC1)NC(c1c(OC)scc1)=O Cc1nn(C)cc1C(O)C(=O)N(C)CC1CCCN(C(=O)CC(F)(F)C2CC2)C1 CC(C)(C(=O)N1CC(CNC(=O)CCc2nc[nH]n2)C1)C1CCCC1 N1(C(c2n(C)c(Cl)cn2)=O)CCC2CN(C(c3cc(=O)n(C)cn3)=O)CC12 C(=O)(CCC(C)N1CCCCC1c1cn(C2CCCCC2OC)nn1)OC C1(C(=O)NCCC2ON=C(C)C2)CCN(C(=O)C(C2CC2)C2CC2)CC1C O=C(O)C(Cc1ccsc1)C(=O)NCCCc1nccn1Cc1ccccc1 C1(CCCN(C(C2(COC)CC(C)(OC)C2)=O)C)CCCCCCC1 O=C1C(CN2CCN(CCc3cnccc3Cl)CC2)c2cc(Br)ccc2N1 c1(C(=O)NC23CCCN(C(C4CCC4)=O)C2C3)ccc(N=c2cc[nH]cc2)cc1 C1(NC(COC)=O)CN(C(=O)CCSC2CCCC2)CC1Cc1c(C)nsc1C C1(CC(=O)NCC2(C(N(C)CC3CC3(F)F)=O)CC=CC2)C=NN(C)C1=O C#CCCC(C(=O)NC(CC(C)C)C(=O)OC)NC(=O)C(C)n1cccn1 O=C1NC(=O)C2(CCCC23CN(Cc2ccc(F)c4cccnc24)C3)N1 Cc1ccc(N)cc1C(N1CC(NC(=O)CN2CC(=O)NC2=O)C(O)C1)=O C(=O)(CCCS(N)(=O)=O)N1CCN(C(c2c(N)cc(F)cc2)=O)CC1CF CN1CN(CCCn2ccnc2-c2cccc(-c3cccc(CN)c3)c2)CC1=O c1(CC(=O)N(CCNC(c2n(CC)ncc2C)=O)C)cc(F)c(F)cc1F C1(O)(C(=O)NCCC)CCN(Cc2ccccc2CSc2cccnc2)CC1 c1(C(N(C2CCCC(N(C(CC(=O)OC)=O)C)C2)C)=O)ncn2c1COCC2 N1(C(C(C)=CCF)=O)CCCCC1CC1C(CCC(=O)N(CCC2CC2)C)C1 C(=O)(C#CC1CCCOC1)NCC1(C)CCN(C(c2c(C)cc(N)cc2)=O)C1 CCCCCCC(=O)N1CCOC(CC(N2CC(CCO)C2)=O)C1 n1(CCC(=O)N(C2CCN(C(C3C(C)C3C)=O)C2)CCO)ccc2cccnc12 c1(N(N2CCN(C(=O)C(C)(F)F)C(CC(F)F)C2)C)ccc2nc[nH]c2n1 N1(C(C(C(CC)C)NC(C)=O)=O)CCC(C)N(C(=O)Cc2cc(CC)no2)CC1 c1(C(c2nnnn2C2CCOC2)NCCNC(=O)OC)csc(Cl)c1Cl C12(CNC(CS(N)(=O)=O)=O)CCCC1CN(C(=O)Cc1cc(C3CC3)on1)C2 c1(C(=O)NCCN(C(=O)CSc2ccccc2)C)cc(F)c(F)cc1N N1(C(c2ccc(C(=O)NC)cc2)=O)CCCN(C(C2CC(CN(C)C)C2)=O)CC1 C(=O)(C(C)CCNC(C1(NC(=O)CC2(O)CCCC2)CCC1)=O)OC c1(OCC(N2CCC(O)(C(C)NC(C(CC#C)C)=O)C2)=O)c(C)cccc1C C12(NC(=O)CCN3CCCC3)CCCCC1N(C(c1cnc3sccn13)=O)CC2 CN1CCN(C(C2CCCN2C)=O)C(C(N2CC(S(C)(=N)=O)C2)=O)C1 N1(C(c2ccn(COC)n2)=O)CCCCCC1CNC(C12COC(CCO1)C2)=O N1(C(c2cnn(C)c2N)=O)CCS(=O)(=O)C(CCNC(C2CC=CCC2)=O)C1 c1(NCC(N2CCC(C)CC2)C(C)C)ccc(=O)n(CC(=O)OC(C)(C)C)c1 N1(C(c2ccnc(O)c2)=O)CCC(NCc2noc(N3CCCCC3)n2)CC1 C1(C)(CNC(=O)NC(c2c(C)noc2C)CC)CC2CC2C1 Cc1c(C(N2CCC(NC(C3C(C)C3(F)F)=O)C2)=O)csc1Br c1(-c2cc(OC(=O)OC)no2)cccc(CN2CCC(C(C)(C)C)(CO)C2)c1 C1(C(N2C(CC)CN(C(c3cc(C)ns3)=O)CC2)=O)CN2CCC1(C)CC2 C1(C(=O)NCC(CN(C(=O)CCCn2cccn2)C)(C)C)CCC(N(C)C)CC1 c1(C(=O)OCC)nc(CNC(=O)NCc2cnc(C(C)(F)F)s2)c(C)s1 C1(C)(C(=O)NCC(CNC(=O)CCSC)OC)Cc2ccc(C)cc2C(=O)O1 c1cnn(C)c1C#N.c1(SC)nc(C(C)NC(C2CC(C(=O)NCC3CC3)C2)=O)no1 c1(OCC)ccc2c(c1C(=O)OCc1c(C)nc3sc(C)cn13)OCO2 C(=O)(C(CC(N)=O)NC(=O)C=Cc1cc[nH]c1)N(CC(COC)O)C c1(-c2cc(C)c(F)cc2)cc(C(N2CC3CNC(=O)C3C2)=O)cc2[nH]ncc12 CCC(CC)CC(F)C(=O)N1CC(C(=O)NCCC(C)CCO)C(F)(F)C1 N1(C(=O)C=Cc2ccncc2)CCC=C(C(=O)N2CCC3CC23)C1 C(=O)(C(=O)N=c1[nH]n(CC(F)F)cc1C)c1ccc(C(CCC)O)cc1 C1(CC(=O)NC(C(N2CC(=C)C2)=O)C2(O)CCC2)CCCOCC1 C(=O)(C1=CCCC1)NC(C)C(CO)NC(C1CCC(CCC(C)C)CC1)=O c1(C(=O)NC2CC(CCNC(c3cc(CCC)oc3C)=O)C2)cnc(Cl)cc1N C1(CNC(CC=C)=O)CC2(CCN(C(=O)C(c3ccc(C)cn3)(F)F)CC2)CO1 CCCC(C(=O)N(CCCNC(C1(CO)CCOC1)=O)C1CC1)OC c1(C(N(CC(C)NC(C2(C#N)CC3CC3C2)=O)CC)=O)ccc2sc(O)nc2c1 c1(OC)cc[n+]([O-])c(C(=O)NC2CCCCC2NC(c2cc(N)ccc2C)=O)c1 N1(C(C(C)NC(=O)OCC)=O)CCC(NC(c2csc(CC)n2)=O)C1C c12nc(cs1)C(C)NC(=O)C2.C1(CC=C)CCC1OC C1(NC(c2ccc(OC)nc2Cl)=O)CC2CC(C1)CN(C(=O)C1CC1)C2 c1(C(=O)NC23CC2CN(C(c2cc(F)n[nH]2)=O)C3)c[nH]c2cccc(Br)c12 C1(CN(C(=O)CSCC(N)=O)C)COCCN1C(=O)CCC(=O)c1ccncc1 C(=O)(C(Cc1cccc(Cl)c1)=NO)NC(C12CC1CN(C(=O)C1=NOCC1)C2)C CC1(C#CC(=O)NC2CC2NC(C2CC(C3CC3)C2)=O)CCCO1 C(CC1=CCN(C(C2CCS(=O)(=O)C2)=O)CC1)NC(=O)CCC1CC1(Cl)Cl C12(C(N3CC(N(C(=O)Cc4cc(C5CC5)on4)C)C3)=O)CC(C1)C(C)(C)O2 C(=O)(CCCS(N)(=O)=O)NC(CC)(CNC(c1cc(O)cc(O)n1)=O)CC N1(C(CC(C)C2CCCO2)=O)CC2C(CNC(c3ncccn3)=O)C2C1 c1(C(N2CC(NC(=O)C(c3ccccn3)O)(CO)C2)=O)ccc(=O)oc1 C(=O)(C1=NOC(C)C1)N1C(C)(CC(=O)NCC(=O)OCC=C)CC1 C(CCCC(CO)NC(=O)Cc1ccnc(O)c1)NC(CCC=CCC=C)=O N1(C(c2n(C(C)C)ncn2)=O)CCCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C(C)C1 C=CC1(C(=O)NC2CCCC2CCF)CCN(C(=O)C(C2CC2)OC)C1 C1(NC(C2CCCO2)=O)CN(C(c2cc(Cl)no2)=O)CC2(CCC2)C1 c1(CNc2scc(-c3c(OCCCC)cccc3)n2)cc(F)c(I)c(F)c1 c1(-c2c(C(=O)NCCC(C)NC(CSCC(=O)OC)=O)c[nH]n2)cccc(Cl)c1 n1(CC(=O)N(CCNC(CN(CCCCCC)C)=O)C)nc(C)c(Cl)c1C C1(O)(CCNC(c2ncc(C3CC3)cc2F)=O)CCCN(C(C2CC(F)C2)=O)C1 C(=O)(C1CCCc2nc[nH]c21)N1CC(NC(c2nc(CC)sc2)=O)C(C)C1 N(C1c2ccccc2CC1NC(C1(F)CCOC1)=O)C(C1(CC(C)C)COC1)=O c1(OC)ccc(C(C)NC(=O)NCCC(Cl)Cl)cc1 c1(C(=O)NCC2(F)CC(NC(c3nc(CCC)oc3)=O)C2)cccc(O)n1 C1(COC)CN(C(=O)C(C)(C)C(C)O)CCN1C(=O)CCc1cccc(Cl)c1 N1(C(CC2(C(=O)OCC)CC2)=O)CC2(COC(CNC(=O)C3=C(Cl)CC3)C2)C1 c1(CC(=O)NCC2C(C)CCCN2C(C2CCOC2)=O)ccc2nonc2c1 c1(C(N2CCOCC(CO)C2)C(=O)NCC)ccc(F)c(SC)c1 n1(CCC)ncc(C(=O)N)c1CC.C(=O)(CSCC)N(CCN)C(C)C C(CC1CCC1)(C(=O)NCCCOCC1CCOC1=O)NC(=O)C=CC1CC1 N1(C(c2n(C(C)C)cnc2)=O)CC=C(CCNC(=O)C2=NOC(C)C2C)CC1 C12CCCN(C1C)C(=O)N2.N1(CCC(C)OC)CCN(C2CC2)CC1.C(C)(C)(C)O C1(CC(=O)NCCC(CNC(c2cccc(OC)n2)=O)O)CCOC(C)(C)C1 C1(C(N2CCSC3(CCC3)C2)=O)CC2(CCN1C(=O)COC1CC1)CC2 N1(C(CC2(NC(CC3CC(=O)NC3=O)=O)CC2)=O)CCC2(C1)CC2(F)F C#Cc1cnc(NCCOCCN(C)C(c2cnn(CCO)c2C)=O)nc1 C1(C(=O)NCC2CCC(NC(c3ccoc3C)=O)C2)(OC)CCCOC1 c1(-c2nc(OC)sn2)cccc2nc(C(N3CCC(N(C)C)CC3)=O)cn12 c1(CC(=O)NCC2CCN(C(COCCC(C)C)=O)C2)ccc2nsnc2c1 c1(C(=O)NC2C3CN(C(CCC=CC)=O)CC32)cc2n(n1)C(C)CCC2 CC1CCC(NC(c2nn(C)cc2Cl)=O)CN1C(c1c[nH]nc1Cl)=O c1(C(=O)NC(C(=O)OCC)COC(=O)CCC2CCC2)c(Cl)ccc(F)c1Cl c1(SC)nn(C)cc1-c1noc(CC(c2cccc(Cl)c2)(C)C)n1 c1(C(=O)NCC(CNC(C2C(C)(C)C2(F)F)=O)O)cc2ncccc2[nH]1 c1(C(=O)NC(CC2CN(C(CC(C)OC)=O)C2)C)cccc(OC)c1 c1(CC)cc(O)cc(O)n1.c12ccc(s1)CC(=O)N(CCO)C1CCN(C1)C2=O C1(C(=O)NCCN2CC3CC3C2)CCN(C(=O)CC2CCCO2)CC1 Cc1ccc(C(C(C)C)NCc2nccs2)cc1OC(C)C C1(CC)CN(C(=O)Cc2nnc(C)o2)CCC1NC(=O)C=Cc1ccnn1C N1(C(CSCc2c(C)nc(C)o2)=O)CCN(C(c2ccccc2)=O)C2CC12 Cc1ccc(Cl)cc1NC(C12CC(NC(c3cccc(Cl)c3F)=O)(C1)C2)=O N1(C(CCOCCOCC)=O)CC2CC(NC(=O)CCC3CC3)CC1C2 c1(C(=O)NCC(C)NC(CN(C(C)=O)C(C)C)=O)noc(C2CCCN2C(C)=O)n1 C1(CNC(C(F)=CC)=O)C(C)CCCN1C(=O)CNC(c1ccoc1)=O C1(C)(NC(COCC=C)=O)CCCCC1C(=O)N(C)CCN(C)CCO c1(C(=O)NCC2CCCC(NC(C=C(C)Cl)=O)C2)ccc([N+](=O)[O-])c(N)n1 N1(C(C(=O)NC)=O)CC(NC(=O)CNc2ccccc2C(N)=O)CC1C C(C)(C)(CCC(=O)NCC1(O)CCN(C(=O)C(F)C(C)(C)O)C1)OC c1(OC)coc(C(=O)NC2CCN(C(c3cnc(S)[nH]3)=O)C(C)C2)cc1=O C=CC(C)(C)C(=O)NC(c1ccc(C)cc1)CNC(c1c(C)n[nH]c1C)=O C1(C(C)NC(=O)CCSC2CCCC2)CCN(C(=O)CCc2cn(C)nn2)CC1 C(=O)(C1=COCCC1)N(C1CCCN(C(c2nnn(C(C)(C)C)c2N)=O)C1)CCO C(=O)(CCC(C)(C)C#N)N(C(C(CC)C)C(=O)NCCC(Cl)Cl)C C(C)(CO)(C(=O)N(CC(C)N(C)C(C)=O)C)OC.c1(SCC)ccc(-n2cncn2)nc1 CC(C)CCC(C)(c1nnnn1CCCF)NCCC(C)CCc1ccccc1 C12(NC(CN(C)C(N)=O)=O)CCCC1N(C(c1nccn1C)=O)CC2 C#CC(CNC(=O)C(O)C1CN(C(=O)CCC2CCCOC2)C1)CC1CC1 c1(C(=O)NC2C(CNC(C3CN(C)C3)=O)COC2)cc2sccc2[nH]1 N1(C(c2c(CC)nn(C)c2)=O)CCC(CO)C(NC(c2c(C)noc2CC)=O)C1 C(=O)(C1=NOC(C)C1)NC(CNC(Cc1c(CC)noc1CC)=O)C(C)(C)C C=CC(CC)CC(=O)NC1CC1NC(=O)CC(C(C)C)c1ccon1 C=C1COCCN(C(n2cc(C3CCC3)nn2)C(=O)NC2CCOC2)C1 c1(C(=O)NC2COCCN(C(=O)CCC3CC3(Cl)Cl)C2)cc2ccccc2s1 C(=O)(C1=CC2(CCOCC2)C1)N1CCCCC(N(C)C(c2cc(CF)on2)=O)C1 Cc1nc2c(C(=O)NCC3CC3NC(C3CN(C(=O)OC)C3)=O)cccc2o1.N(C)C C1(O)(CNC(=O)C(F)=CCCF)CCCN(C(=O)Cc2cncc(O)c2)CC1 C1(C(N2C(CNC(=O)Cc3sc(O)nc3O)CCC2)=O)Cc2cccc(F)c2O1 N1(C(c2c(C)ccnc2O)=O)CC2(CCC(CNC(=O)Cc3cccnc3)O2)C1 C(=O)(C#CC(C)(C)C)N(C(C)CCNC(c1sccc1Cl)=O)C C(=O)(C1=NOC2COCC12)NCCCCC(C)NC(c1[nH]cc(C)c1)=O N1(C(CSC)=O)CC(NC(C2COCCC2(F)F)=O)CC1(CC)CC c1(CC(=O)N(CC)CC2CCCN2C(=O)C(CN(C)C)N(C)C)cccc(Cl)c1 N1(C(CC(CNC(C(CC)CN(C)C)=O)C2CCC2)=O)CC2(C1)CN(C)C2 c1(C(=O)OCC)cc(OC)cc(NCP(C)(C)=O)c1Cl C(=O)(C(CC(F)F)NC(c1ncccc1N)=O)N1CC(CC(C)C)OCC1 C#Cc1cc(C(N2CC(CCNC(c3ccccc3C)=O)(OC)C2)=O)ccc1C C1(C(=O)OC)CC2(CCOCC2)CN1Cc1cccc2c1OC(C)(C)C2 C1(NC(C(C)C2CCCC2)=O)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1 Cc1cc(C(N2CC=CC(NC(c3n[nH]cc3Br)=O)C2)=O)ncc1C#N N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2(C1)CN(C(c1sccc1Cl)=O)CCO2 CCCC(F)C(=O)N1CCCC1C1CCN(C(C2CCOC2)=O)CC1 C(=O)(CC(C)C(F)F)N1CCC(C(CNC(COCC#C)=O)(C)O)CC1 Cc1c(C(N2CC(NC(C3CC34CC(C)(C)C4)=O)C(O)C2)=O)cncc1N c1(C(=O)NC(COC)CNC(=O)C(C)C2CCCC2)ccnc(C)n1 N1(C(CCCOCC=C)=O)CCN(C(c2cnn(CC(C)C)c2)=O)C(CF)C1 N1(C(C(=O)NCC)=O)CCCC2(C1)CN(C(=O)C(C)CN1CCCC1)C2 C(CC(C)(C)C)(C(=O)NC1COC(C(F)F)C1)NC(C(c1ccncc1)C)=O C(c1nc(C)cs1)=CC(N1CC(C(C)(C)O)(CNC(CC(C)OC)=O)C1)=O CC(C)C(C(=O)NCC(C)CNC(=O)COCCSc1ccccc1)NC=O c1(C(=O)NCC(=C)CCNC(=O)CC(=O)NC2CC2)cc(NC)nc(C)c1 c1(CONC(=O)CC2CCCN2C(=O)CN2CCOCC2)cccc(F)c1 Cn1cc(CNC(C23CC(F)C2C3)=O)c(C(F)F)n1 N#Cc1ccc(-c2ccc(NC(C34CCCC3CCC4)=O)cc2)nc1 C1(CC)(CO)CCCN(C(=O)COC2CCN(C(C3CCCC(O)C3)=O)C2)C1 n1(C(C)C(=O)NC(C)CN(C)C(c2cnc[nH]2)=O)cnc2ccccc12 C1(CNC(CCOCC)=O)COCC1NC(=O)CSCCC1CCCC1 C(C)(N=c1nc(N2CC(NS(C)(=O)=O)C2)c2c([nH]1)CCC2)c1n(CCC)ncn1 C1(CNC(=O)NC(c2nc(C)sc2)c2ccccc2)CN(C)CCC12CC2 C12(NC(CCCCC=C)=O)CCCCC1N(C(=O)C=Cc1ccnn1C)CC2 C(=O)(C(O)CCCNC(C1CCC2(CC1)CC2)=O)N(C1CCCC(O)C1)C Cc1nc(Cl)nc(N2CC3CC2CCC3NC(C2(C)CCS(=O)(=O)CC2)=O)c1F N1(C(CCCCCCC)=O)CCC(NC(=O)CCC2CCCN2C)C(CO)CC1 CCC(CC(=O)NC(C(=O)NCC(c1ncc[nH]1)C)c1ccoc1)C(F)F C(=O)(CCCn1cccn1)NC(c1cc(I)on1)(C)C C(=O)(C(CC(C)C)C(C)C)NCC1CCCN(C(C2CC(CC)C2)=O)C1 c1(C(=O)NC(CNC(C(CC=C)(C)CC)=O)COC)cc(C)c2occc2c1 c1(OC)nsc(OC)c1C(N1CCOC(CNC(=O)CN(S(=O)(=O)CC)C)C1)=O N1(CCCC(=O)NCC(CNC(C2C(C(N)=O)C2)=O)O)C(=O)CNC1=O c1(C(N2CCC2CNC(C2CCN(C)C(C)C2)=O)=O)cc(F)c(N)c(F)c1.CO c1(C(=O)NCC(CC=C)NC(CC=C=C)=O)cc(F)c(Br)c(F)c1N c1(-c2n(CCOCC)nc(Cc3ccc(OCC)cc3)n2)cc(OC)ncc1Cl c1(-n2cc(C3CN(C(CSCC(=O)Nc4cccs4)=O)C3)nn2)cncc(Br)c1 C(=O)(C(C(C)(C)C)N(C)C)NC(C(C)NC(CCCCNC(C)=O)=O)(C)C C1(C(N(C(C(=O)NCC(C)(C)C)C2CC2)C)=O)CC2CC2C1 C(C(C)(C)CC(=O)N1CCC(NC(=O)COC(C)C)C2CC12)OC c1(OC)cccnc1C(c1nnnn1C)N(CC(N1CCOCC1)C)CC c1(SCC(C=C)CC)nc(Cl)c(C)cc1F N1(CC(N2CCC(N(C(CCN(CC)CC)=O)C)C2)=O)CCNC(=O)C1 Cc1nn(C)cc1C(N1CC(F)CC1C(=O)Nc1cn(C)nc1C(F)(F)F)=O Cn1c(=O)c2nc(CN3CCCC3C3CCCN(CCO)C3)[nH]c2n(C)c1=O c1(CC(=O)NCC2CN(C(CCCC)=O)CC2(F)F)nn(C)cc1[N+](=O)[O-] C1(CC)CN(C(c2cn(CCNC(=O)C(F)F)nn2)=O)CC(=O)N1 c1(OC)ccc(OCC(N2CCC=CC2CNC(=O)C=Cc2cocn2)=O)cc1 C1(NC(C2(C(=O)OCC)CC(=O)C2)=O)CC2CC1CC2C(=O)NC1CC1 C1(CCC)CN(C(=O)CC2(C)CCCCO2)CCN1C(=O)CN1CCCCC1=O C1(NC(=O)Cc2cccc(Br)c2)COCCN(C(C2(C3CC3)CCC2)=O)C1 c1(OC)cc(C(=O)NCC(O)CNC(=O)C(C)O)c2ccccc2c1 N1(C(CCN(C(C)=O)C)=O)CC(NC(=O)CCC(N)=O)C2CC12 N1(C(c2c(CC)nccn2)=O)CC(NC(=O)C=Cc2ccccc2)C2(CCC2)C1 c1(C2CCN(CCCC)C2)cc(NC(=O)CCCCNC(=O)NC)ncn1 c1(C(N(C(c2ccc(Br)s2)C(=O)NC)C)C)nc2ccccc2s1 N1(Cc2nc(=N)o[nH]2)CCc2ccc(C(F)(F)F)cc2C1 c1(CNC(=O)CC2C=CS(=O)(=O)C2)cc(Br)c2c(c1)OCCO2 C1(CC(=O)NCc2nc(C)c(C)s2)C2CCCC2N1C(C1CCC(C)(O)CC1)=O c1(NCc2ccc(C)cc2C)cc(=NCCc2ccc(S(C)(=O)=O)s2)[nH]c(C)n1 C1(NC(COC)=O)CCN(C(C2CCCOC2C)=O)CC1C C(=O)(C1=CS(=O)CCC1)N(CC(CC)NC(c1ccn(CCC)n1)=O)C C(=O)(C(C)(F)C(=O)N1CC(NC(c2cnc(C(F)(F)F)nc2)=O)CC(F)C1)OC CC(CC(=O)N(C(C)CCNC(C1(C)CN(C)C1)=O)C)n1ccnc1 C1(C(C(=O)NC2C(CCCC)CCC2)C)CCN(C(c2cc[nH]n2)=O)CC1 C=CC(CCC)CC(=O)NCCN(C(=O)CCC(=O)c1ccccc1)CCOC C12(NC(c3c(C)nc[nH]3)=O)CC(CNC(C3CC4CCC(C3)C4)=O)(C1)OC2C c1(C(N2CCN(C(CC3(NC(C)=O)CC3)=O)C(CO)C2)=O)ccc(Cl)c(C)c1O C(=O)(CCC(C)CC)N(C1CCN(C(c2c(C)[nH]c(C)c2C)=O)C1)CC#C C(=O)(C(C)C(C)(C)C)N(CC(=O)NCC1(CC)CCC(=O)N1)CCC C1(NC(=O)OC(C)(C)C)CC2(CCC2NC(c2cccs2)(C)C)C1 CC1=C(C(=O)NCC(C2CCCCC2)NC(=O)CC2CC3(CC3)CO2)CCC1 C1(C(N2C(C(=O)Nc3ncccc3Br)CCC2)=O)CCCC2CCCCC12 N1(C(C2CCN(c3n(C)ccn3)C2)=O)CC2CC(NC(=O)C(C)(C)CF)C(C2)C1 c1(OC)ccc([N+](=O)[O-])c(CN2CC(C(N3CCCC(C)(O)CC3)=O)C2)c1 C1(C(=O)NC2(CC(N3C(COC)CCC3)=O)CC3(CC3)C2)CCC2(CCC2)O1 C(C)(CN=c1cccc(S(=O)(=O)NCc2nccn2C)[nH]1)OCCCC N1(C(CCC=C=C)=O)CC2CCCC1CN(C(=O)C=CC(C)(C)C)C2 N1(C(C(CC)C2CCCCC2)=O)CCC(NC(=O)Cc2cnoc2)CC1C C1(CNC(CC(CC)C)=O)CN(C(c2ccnc(C)c2)=O)CCC12CCC2 CC1(C)NC(=O)CCC1CN1CCS(=O)(=O)CC1C(F)(F)F O=C1CCC(CC(=O)NC2C3CCN(C(c4ccsc4Cl)=O)C23)CN1 C1(C)(NC(C2N(C(C(C)=C3CCC3)=O)CC2C)=O)CCC(=O)N(C)C1 C1(CCNC(=O)Nc2ncc(-c3ccccc3)s2)CCCCCC1 c1(OC)ccc(C(=O)NC(CN(C(=O)C(C)c2ccsn2)C)(CO)CO)nc1 CC(C)C(C#N)C(=O)N1CCC(C(N2CC(OC(F)F)C2)=O)C1(C)C c1(CC)ncoc1C(=O)NC(C(N1CCC(CN2CCCC2)C1)=O)C1CCCO1 c1(C(=O)OC)ccc(C)c(C(=O)NC(CNC(C2CCCS2(=O)=O)=O)C2CC2)c1 N#Cc1cccc2c1CN(Cc1nc3ccccc3n1C(F)F)CC2 C12(C(=O)NCC3N(C(C4ON=C(C)C4)=O)CCCC3)CCCC1CCC2 CC(c1ccccc1F)=CC(=O)NCC#CCNC(C1CC1[N+](=O)[O-])=O C(C)(C(=O)NOCC1(C)CC1)NC(C(C)n1cccn1)=O [N-]=[N+]=NC1CN(C(C2(CC(F)F)CC2)=O)CC1NC(C1CC12CCOCC2)=O c1(C(N2CCC(C(N(C(C)C)CC)=O)C2)=O)sc(Br)cc1Cl c1(C(N(C2CC(NC(CC=C(C)C)=O)C2)C)=O)ccc(Br)cc1C#N C(=O)(CCCCCCCCBr)N1CC2CN(C(c3c(C(N)=O)cccc3)=O)CC21 CN1CC(NC(C2CCCNC2)=O)CC1=O C1(C(=O)NCCC2(C)CCN(C(C3C(C)C3)=O)CC2)Cc2ccccc2C1 C1(C(=O)NC(C23CCCC2C3)C)(CNC(C2COCCO2)=O)CCCCC1 Cc1cccc(C(N2CC(NC(=O)Cc3nc(C)c(C)s3)C3CC23)=O)n1 c1(CCC(N2C(CN(C(c3cc(CC)no3)=O)C)CCC2)=O)ccc(C)c(C)c1 C(C1=NOC2CN(C(=O)CCOC(C)C)CC12)NC(Cc1c(C#C)cccc1)=O Nc1ccc(C(=O)NCC2(NC(c3cccc(OC4CC4)c3)=O)CC2)cc1Cl c1(C2C(C(N3CC(F)CC3CNC(C3(F)CC3)=O)=O)C2)c(F)cccc1Cl c1(OCC)ccc(C(=O)NC2CN(C(=O)C=NOC)CCC2C(F)(F)F)cc1N N1(C(C(CN(C)C)c2ccccc2)=O)CCC(C)(CNC(=O)OC(C)(C)C)CC1 c1(OC)cc(C(=O)NCC2CCN2C(C23CCC(CC2)C3)=O)c2c(c1)CCCC2 C1(NC(c2scc(C)c2C)=O)CN(Cc2ccc(C#N)cc2O)CCC1(F)F c1(C(=O)NC(C)C(C)NC(c2ccc(Cl)o2)=O)csc(C(C)(C)C)n1 CCCCCCC(C)CC(=O)NCC1CN(C(=O)CN=S(C)(C)=O)C2(CCC2)C1 Cc1cc(C)c(C(N2CC(NC(c3ccc(SC(F)(F)F)cc3)=O)C2)=O)[nH]1 c1(C(=O)NC2C(C)(C)N(C(C3CCSCC3)=O)CC2)nc2cccnc2s1 Cc1noc(C)c1C(C)(C)C(=O)OCCCOCCOCCOCCNC(C1(F)CCC1)=O.O.OO CCCCC(C(=O)NCc1ncc(CC)[nH]1)NC(c1cnc(O)c(F)c1)=O CC(C)(C#N)CC(=O)NCCC1(O)CN(C(=O)CCC2CC(C)(C)CO2)C1 C1(O)(C(=O)NCC2(C)CCC(NC(CC=C(C)C)=O)CC2)CCC(C)(C)CC1 C12(C(=O)NC(CC)(CNC(C3CC3(C)C(F)F)=O)CC)CCCN1CCC2 n1(CC)ncc(Cl)c1C(=O)N(C)CCNCc1cn(Cc2cccc(F)c2)nn1 CN1CC(C(=O)NCC2C3CN(C(c4csnn4)=O)CC23)OCCC1=O C1(C(N)=O)COCCC12CNC(C(C1CCN3CCC1C3)=O)C2 C1(C(N(CCCNC(=O)C(c2ccc(F)cc2)CO)C)=O)Cc2ccccc2N1 N1(C(c2ccc(C#C)cn2)=O)CCC2(CCCN2C(=O)CCc2ccccn2)C1 c1(C(N(C2(C(=O)NC(C)CCN3CCCC3)CC2)C)=O)cc(F)c[nH]1 C12(C(=O)NCC3(OC)CN(C(c4cc(Cl)ncc4F)=O)C3)CC(C)(C1)OC2C C12(C(N3CC4C(N(C(=O)CC5CSCCS5)C)C4C3)=O)CCC(CC1O)C2 C(CCC(O)C(=O)NCc1cc(C(N)=O)no1)NC(Cc1c(C)ocn1)=O C1(NC(C2CC(SC)C2)=O)CCC12CCN(C(=O)C(C)Oc1cccnc1)CC2 CC(C)C(C#N)C(=O)NC1(C)CC(C(=O)NC2CCC3CC2CO3)C1 CC(C)CCCC(C)CNC(=O)CNC(C1CC2C=CC1C2)=O N1(C(C(c2ccccn2)C)=O)CCOCC(NC(c2sccc2CO)=O)C1 C=CC(C)(CC)C(=O)NC1(C2CN(C(c3ccc(CO)cc3)=O)C2)CC1 c1(OC)cncc(C(N2CCCC2NC(=O)C(=O)Nc2ncc[nH]2)=O)c1 C1(N(C(CCCC)=O)C)CN(C(C2COC(=O)C2)=O)CC1(C)C C1(C#N)(OC)CC(C(=O)N(CC(O)CN(C)C(c2cc(C(N)=O)[nH]n2)=O)C)C1 N1(C(Cc2cc(OC)ncc2)=O)CC2CCC1C2NC(c1cc(C)oc1C)=O N1(C(c2cnn(CC)c2C2CC2)=O)CCOC(C)(CNC(=O)C(F)OC(F)(F)F)C1 c1(N(C(Cc2c(C)nc[nH]2)=O)C)cccc(F)c1 c1(C(=O)NCC2CCCC(NC(C3(OC)CCC3)=O)C2)cnc2occc2c1 c1(C(=O)NCC(CNC(C2(C)CCN(C)CC2)=O)CO)cc2cccnn2c1 c1(SCC(=O)NC2CCN(C(c3ccccc3)C)CC2)ncc2c(n1)CCC2 c1(C(=O)NC2(CN(C(=O)C3=CC4CCCC34)C)CC2)ccc2c(n1)CCC2 Cc1nccc(C(=O)NCC2CN(C(C3CCOC3C)=O)CC2C(F)(F)F)n1 C1(C)(NC(C(c2ccccc2)C)=O)CCN(C(c2ccc(C(F)(F)F)s2)=O)CC1 C1(NC(c2ccc(Oc3ccc(C)cc3)nc2)=O)CCC(C2CC2)C1 C(C(CC)(CC)NC(c1cncn1C)=O)NC(C1C(CC)OCC1)=O C12(C(=O)OC)CCCCC1CN(S(=O)(=O)CC13CCCC(C)(CO1)C3)C2 C1(C(C)NC(Cc2cn(CC)nc2)=O)CN(C(C2(n3ccnn3)CC2)=O)CCO1 c1(C(=O)NC2CCC(NC(CCn3ncc(C)c3)=O)C2)noc(C2CC2)c1C c1(OC)cnc(C(F)(F)F)[nH]c1=NC1CCC(C(N2CCC(F)C2)=O)CC1 C(=O)(C(C)(C)C(F)F)NC1C=CC(CNC(CC(C=C)C)=O)C1 C12(NC(C3CC(C)(C)OCC3)=O)CCCC1N(Cc1ccc(C(F)F)cc1)CC2 N1(C(c2c(C)noc2)=O)CCCCC(C(=O)NC2CCN(C)CC2C)C1 CCC(O)C(C)C(=O)NCCOC1CN(C(c2cc(C(F)(F)F)cs2)=O)C1 N1(C(C(CCN(C)C)NC(CCc2c(C)cccc2)=O)=O)CC(O)CC(O)C1 N1(C(c2ccc(N(CCC)CC)cc2)=O)CCN(C(=O)CCCOC)C(C)C1 C1(NC(c2ccn(C)c2)=O)CC2CC(NC(C3(O)CCSC3)=O)C1C2 CC(C(=O)NNC(=O)COc1ccc(N2CCN(C)CC2)cc1)c1ccsc1 N1(C(CCC=C)=O)CCC2(COC(CNC(=O)CS(=O)(=O)NC3CC3)C2)C1 C1(CNC(c2cc(C(N)=O)co2)=O)CC(CO)NC1.c1(SCC(=O)OC)nncs1 Cn1nccc1C(C(N1CC(O)(c2cnn[nH]2)C1)=O)NC(=O)CO C(CC(C)(C)CNC(=O)CC(CC1CC1)NC(C1CCC(N(C)C)C1)=O)OC N1(C(Cc2c(C)ocn2)=O)CCN(C(=O)CCc2cc(Cl)cs2)CC1CC(F)F N1(C(C(C)OC)=O)CCOC(CN(C(=O)CCC(C)OC)C)C1 c1(CC(=O)NCC(CO)NC(CCOC)=O)csc(C(C)SCC)n1 C(Cc1cnc[nH]1)(C(=O)NC1COC(=O)C1)NC(C(C)=C(C)C)=O c1(NC(n2cc(C(=O)NCC(C)SC3CCCOC3)nn2)=O)ncnc2c1CCC2 c1(SC)cc(C(N2CC3C(CN(C)C(c4cccn4C)=O)C3C2)=O)c(C)o1 C1(CCC(=O)NCCN(C)C)CCCN(C(=O)Cn2cccn2)C1 CCCCCC(O)CC(=O)N1CC(NC(=O)Cc2cccc(OC)c2)C(F)C1 c1(C(=O)NCC2(F)CC(CNC(CC(C)F)=O)C2)cn(C)c(=O)cn1 C(=O)(CCC(C)C(C(=O)NC(C)C(=O)NC1CC1)N1CCCC1c1ccco1)OC c1(NC2N(c3nc(C(=O)OCC)c(Br)cn3)CC2)cc2c(cc1Br)OCCO2 Cc1nc(C(=O)NCC23CC2CN(C(C2C(C(F)F)C2(C)C)=O)C3)c(C)n1C c1(OC)cc(N)ccc1C(=O)NCC#CCNC(c1sccc1F)=O N1(C(c2cc(CCC)on2)=O)CCC(CC(=O)NC(C)C(C)O)CC1 [N-]=[N+]=NC1CCC(NCc2cnn(-c3ccccc3Br)c2)CC1 CC1CCC(Cl)=C(C(=O)NCC2CC2NC(c2ccc(-c3ccccn3)s2)=O)C1 C1(C(C(=O)NC(c2cn(-c3ccccc3)nn2)C)O)CCOCC1 C(=O)(CC(CC1CC1)NC(c1cc(C(C)C)[nH]n1)=O)NC(CCC)CC C1(C(=O)NCC2N(C(CN3CC(C)C3)=O)CCN(C)C2)CC2(CCCC2)CO1 c1(N2CC(C)C(CO)C2)nc2ccc(Cl)cc2c(=NC2CCCC2)[nH]1 C1(NC(CCNC(c2occ(C)c2)=O)=O)CCN(C(=O)COc2ccccc2)C1C c1(C(N2CCC(NC(c3nccc(OC)c3)=O)CC2C)=O)cc(F)cc(N)c1F CC1(CNC(=O)CNc2cnccn2)CCCN(C(=O)CC23CCCC2C3)C1 Cc1cc(C(N2CC(C)(c3cn(-c4ccc(F)cn4)nn3)C2)=O)nnc1C c1(C(N2C(CNC(C(C)OCC)=O)CC3CC32)=O)ncc2c(F)cccn12 CCCCC(CC)CC(=O)N1CCCC1(C(=O)NCc1ncsc1C)C(C)C C1(NC(c2c(C)ccnc2)=O)CN(C(=O)CCS(C)(=O)=O)CC2(CCC2)C1 N1(Cc2ncc(C(C)C)s2)CCC(C)C1c1cn(-c2ccccn2)nn1 c1(CC2N(CC(n3cccn3)C)CCCC2)cc(S(N)(=O)=O)cn1C c1(CC)nc(C)n(C)c1C(N1CCCC(N(C(c2cnn(CC)c2)=O)CC)C1)=O C#CCC(CCc1ccccc1)N(c1cccs1)C(=O)CC1CCC(C(C)C)CC1 N1(C(CC=CC)=O)CCCCCC1CNC(c1ccc(OC(C)C)cc1Cl)=O c1(C(N2C3C(NC(=O)C(F)=CC4CC4)CC(C3)C2)=O)ccn2c1CSCC2 C#Cc1cc(C(=O)NC2(CNC(=O)CC(C)(C)N(C)C)CCOCC2)ccc1Cl c1(OC)ccc(C)c(NC(=O)NCc2ccn(CC(C)C)c2)c1 CCCC(O)C(=O)N1CCN(C2CCN(C(=O)CC3CC3)C2)CC1 c1(C(=O)NC(CC=CC)C(=O)NCCSC)ncnc(O)c1F c1(C(=O)NC(C(C)NC(c2onc(CC)c2C)=O)C)n[nH]c2cc(Cl)ccc12 C(=O)(C(C)(C)S(C)(=O)=O)NC1C=CCN(C(CC2C(C)=NOC2=O)=O)C1 c1(C(=O)NC(CC)CNC(=O)CNC(c2cccs2)=O)cc(Cl)cnc1OC C(c1ccc(F)cc1F)=CC(N1CCCC(CNC(C(C=C)O)=O)CC1)=O C(=O)(CC(C(C)(C)C)NC(=O)C=Cc1ccc[nH]1)NCc1ccc(C#C)cc1 N1(Cc2c(C)nc[nH]2)CCC12CCN(S(=O)(=O)CC#N)CC2 C(=O)(C1=CCC(C)(C)CC1)N1CCN(C(C(CSC)O)=O)C(C(C)(C)C)C1 c1(CC(=O)NC2CCC(NC(CCOCCC)=O)C2)coc2ccccc12 c1(C(=O)NCCC(=C)CNC(C)=O)cncc(OCCC(C)OC)c1 c12ccc([nH][nH]c(=O)[nH]1)nc2.C1(C(=O)OC)CCC(C)C1 Nc1ccc(Cl)cc1C(N1CCC(NC(C2(Br)CC2)=O)CC1C1CC1)=O C1(C(N2CC(C)C(NC(=O)Cc3ccc(C#N)cc3)C2)=O)CC2C=CC1C21CC1 C1(NC(C(C)C)=O)CN(C(c2cnn(-c3ccccc3)n2)=O)CC2CC12 c1(OCC(=O)NCC(CNC(c2cc(CO)n(C)n2)=O)OC)cc(F)ccc1F C(=O)(CCCCCS(N)(=O)=O)NCC1CC(NC(C(C)Oc2cccnc2)=O)C1 Cc1ccc(OCC(=O)NC2CCC(F)(CNC(=O)C=Cc3cscn3)C2)cc1 C(=O)(C(F)(F)COC)N(CCNC(C1C(C)C1C)=O)CC c1(C(=O)NCCCCCNC(c2ccc(C)cc2Cl)=O)c(F)ccc2occc12 CCCC(C)C(=O)NCCC(O)CNC(c1nc(-c2ccc(Cl)cc2)oc1C)=O CC1Oc2c(C(=O)NC(CO)CCC(C)(C)C)cccc2C1C c1(C(=O)OC)cc(NC(N2CCCC(C(F)(F)F)CC2)=O)cc(Cl)c1 N1(C(c2n[nH]c(C)c2F)=O)Cc2occ(C(=O)NCc3ncc(F)cc3F)c2C1 C1(C(=O)NCc2ccncc2)(CNC(C2C(C(C)(F)F)C2)=O)CCCO1 C1(CNC(=O)CCn2cncn2)CN(C(C2CCC(=O)O2)=O)CC1(F)F C1(C(=O)NC(C(C)C)CNC(c2nnc(C(C)(C)C)s2)=O)(CO)CCCCC1 Cc1ccc(OC(C)C)cc1-c1nc(C2C(c3ccccc3)C2(C)C)no1 N1(C(CP(C)(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)CCNC(N)=O)C3 C(=O)(C1=CC2(CCN(C(C3(CC)CCCCC3)=O)C2)C1)NC1CC1c1ccco1 C1(C(=O)NC2CN(C(c3ccn4ccsc34)=O)C2)Cc2ccccc2CO1 c1(OC)cc(C)nc(N2CCCC(NC(=O)CCc3ccc(O)nc3)C2)n1 Nc1ccc(-c2cn(-c3cccc(C(=O)Nc4ccccc4)c3)nn2)cc1F c1(C(N2CCN(C(C(CC(CC)C)C)=O)CC2)=O)cc2ccc(O)cc2[nH]1 c1(OC)ccnc(N2CCOC(C(=O)NC(c3ccno3)C)C2)n1 c1(C(N2CCCC(c3cn(CCCOC)nn3)C2)=O)cc(S(C)(=O)=O)ccc1F c1(CC(N2CCC(NC(C3C4CCC3CC4)=O)C2)=O)nccc2ccccc12 C=C(C)CC(C(=O)OC)NC(=O)CC12CC1CCN2C(=O)CCC=C(C)C C1(O)(CN(C(C2CN(C(C)=O)C2)=O)C)CCN(C(=O)CCCC2CCC2)C1 N1(C(CC(=O)OC)=O)CC(=O)NCC1C(=O)NCC1CCOCC1(C)C Cc1cc(Br)cnc1C(=O)NC1CC1CNC(c1cccc(=O)o1)=O Cc1cc(C2CCN(C(=O)C(N3CCN(C(C)C)CC3C)=O)CC2)cc(O)c1.N c1(C(N(C)CCNC(=O)C(C)(Cl)Cl)=O)cc2n(c1)CCOC2 Cc1ccc(C(=O)NCC(C)(C)NC(=O)C(C)(C)CN2CCN(C)CC2)c(C)n1 c1(CCCCNC2CCCC(OC)C2)cn(C2CCc3c(Cl)cccc32)nn1 O=C(NN1CCCCC1=O)c1coc2ccc(Cl)cc12 Cc1nc2ccccc2cc1C(=O)N(C1CCCN(C(C2(C(C)C)CC2)=O)C1)C c1(C(N(C2CCCN(C(Cc3cn(CC)nn3)=O)C2)C)=O)cn2c(n1)COCC2 Cn1ccc2cc(NC(C3(CNCc4cc(Br)c(F)cc4Cl)CC3)=O)ccc12 C1(N(C)C)(C(=O)NC2CCCC(N(C)C(C3(C)CC(F)(F)C3)=O)C2)CCCCC1 c1(OC)ccc(F)cc1C(=O)C(=O)N(CCCN(C)C(c1cocn1)=O)C C1(C(=O)NC2CCC(C3CC3)C2)(CC)CCN(C(c2cn[nH]c2)=O)CC1 C1(C)(C(=O)Nc2ccc(CN(CCC)CCC)cc2)CCN(C(c2csnn2)=O)C1 N1(C(c2cc(C)c(Br)s2)=O)CCN(C(=O)CN(C)C)CC12CC2 C=Cn1nncc1C(N1CCCC(C(=O)NCCNC(=O)C(C)C(F)F)C1)=O O=S(=O)(c1ccc(NCc2cc(C(F)F)no2)c(F)c1)N1C2CCC1CC(O)C2 N#CC1=C(C(=O)NCCN2CCN(C(c3onc4c3CCCC4)=O)CC2)CCC1 c1(C(C2(C(F)(F)F)CCN(Cc3ccccc3OC(F)F)C2)=O)cccc(Cl)c1O C1(F)(CNC(c2c(C)oc(C3CC3)n2)=O)CCCN(C(c2cnsc2C)=O)C1 CC1(C#CC(=O)N2CCN(C(=O)CCC3CCC3)CC2C2CC2)CCCO1 CC1(C(N2CC(CO)(NC(c3cnc(C(C)(C)C)[nH]3)=O)C2)=O)CC2(CC2)C1 CC1CCCN(C(=O)C(=O)NC2(C)CC(CNC(=O)C(C)c3ccsc3)C2)C1 C1(Cc2n(Cc3cccc(F)c3)ccn2)CCCN(CCC2=CCCCC2)C1=O C1(NC(c2c(OC)cncc2)=O)CCC2CCN(C(c3csc(Cl)n3)=O)C1C2 Cc1cc(CCC(=O)N(C2CC2)CC2CCCN(C(c3ccon3)=O)C2)c(C)s1 c1(N(C)C)ccc2cc(C(=O)NCC3C=CCN3C(=O)C3=CCOC3)ccc2n1 c1(C(=O)NCCC(CO)SC)cc(Br)cc([N+](=O)[O-])c1N CC(C)(C)C(CC(=O)N1CCC(OC)C1)NC(C1(CO)CCOCC1)=O c1(-c2scc(C(=O)NC3CN(C(CCOCC)=O)C3)n2)cccc(C)n1 C(C)(CN=c1[nH]cc2ncnc-2[nH]1)OCC(NC1c2cccc(C)c2OCC1)=O CCCC(CNC(c1cn(CC)cn1)=O)C(=O)NC1CCSC1 c1(C(=O)OC(c2cccc(-n3cccn3)c2)C)ccc2ccn(C)c2c1 CCCCC(C)(CO)NC(=O)C(O)C1CN(C(=O)CCCC(C)C)C1 C1(C(N2CCC(c3cn(-c4cccc(I)c4)nn3)C2)=O)(OC)CS(=O)(=O)C1 c1(CC(=O)NC2COCC2C)ccc(O)cc1.C1(Cl)(C(=O)NCC2CC2)CC1 N1(C(CCCCC#C)=O)CCCCC2(CCN(C(C3(O)CC3)=O)C2)C1 C(C)(CCN=c1[nH]c(Cl)ncc1[N+](=O)[O-])NC(CC1CCC(C(C)C)CC1)=O c1(C(=O)NC(CCC)CC(=O)N2CCC=C(Cl)C2)ccc2ccoc2c1 c1(N2CCN(C(=O)OCC)CC2)ccc(S(=O)(=O)N2CC3COCC3O2)cc1 N1(C(c2c(OC)ccc(C)c2)=O)CC2CCC(C1)N2C(C1CN2CCCN1CC2)=O CC(C)S(=O)(=O)c1ccc(Cl)c(C(N2CCc3cccc(F)c32)=O)c1 N1(CC)CC(C(=O)N(C)CC2CCCN2C(=O)C=Cc2cncs2)NC1=O c1(NC(C2CCC3(CN(Cc4cccc(I)c4F)C3)O2)=O)ccc2n[nH]cc2c1 N1(C(c2c(CCC)occ2)=O)CC(NC(C2CN(C(C)C)C2)=O)C(C)C1 c1(NC(c2scc(NC(=O)Cn3ccnn3)c2)=O)ccc(-c2nc(=O)o[nH]2)cc1 Cc1ccccc1C(=O)NCC(C1(O)CN(C(=O)C(F)CC2CC2)C1)(C)C c1(CN2CCC(N(CCC#N)C(c3cn(CCCC)nc3)=O)C2)ccc(C)cc1 C(=O)(C(=O)C(C)C)NC(c1cn(C)nn1)C(=O)NC(c1c(C)ncs1)C C1(C(=O)NC(C)C(C)(C)NC(c2cccc(C3CC3)c2)=O)COCCC1(F)F c1(C(N2CC3CN(C(CCCCC=C)=O)CC32)=O)cc2cccc(Cl)c2o1 C1(C(N2CC(n3cc(CC(C(C)C)O)nn3)C2)=O)CCCCCC1.C12CC(C1)O2 c1(OC)n[nH]c(C(=O)N(C2CCN(C(c3cnc(C(F)F)nc3)=O)C2)C)c1Cl c1(C(=O)NCCCCCCNC(=O)CC2CC(F)C2)cn2ncccc2n1 N1(C(CNC(N(C)CC2CCCC2O)=O)(C)C)CCCCC1 C(=O)(C(F)(F)CC=C)N1C2(n3cc(COc4nc(COCC)[nH]n4)nn3)CC(C1)C2 c1(C(NNC(=O)NCC2CN3CCN2CC3)=O)ccc2c(c1)OCCO2 N1(C(=O)OC(C)(C)C)CCN(c2cc(C(N3CC(O)CC3C(F)(F)F)=O)ns2)CC1 N1(C(c2ccc(C)s2)=O)CC2(C(=O)NC(C3CCCO3)C)CC1C2 c1(NC(C2CC(NS(=O)(=O)C3CCC3)C2)=O)nc(Cl)c2ccnc-2[nH]1 N1(C(Cc2c(C)ccnc2)=O)CCC2CC1CN2C(c1[nH]nnc1C)=O CC(Cc1cnn(C)c1)C(=O)NCCOC(C)(C)CNC(C1(F)CCC1)=O Cc1cccc(-c2ccc(C3CCCN(C(c4snnc4C)=O)C3)s2)c1 N1(C(CC=C)=O)CCCC1C(C)NC(c1ccoc1CC)=O C(=O)(CCCS(C)(=O)=O)NCC1CC(F)(CNC(c2c(C)nc(C3CC3)o2)=O)C1 Cc1cccc(CCC(N2CCC(NC(c3cnoc3C)=O)C(C)C2)=O)c1Br CC1(O)CCN(C(C2CC(CCNC(=O)C=CC3CCCC3)C2)=O)C1 c1(C(=O)NC(CN(C(C=C(C)Cl)=O)C(C)C)C)cccc2c(C)[nH]nc12 c1(C(N(CCc2ccc(C)cc2)C)=O)cccc2c1C(C#N)C2 c1(C(=O)NCC(CC=C)NC(c2ccc(C=C)cc2)=O)cc(F)ccc1C(C)C c1(CNC(CN2CCC(OC)C2)=O)cc(C)c(C(=O)NCc2cnn(CC)c2)o1 c1(NC(C23C(CN(C(c4ccccc4I)=O)C2)C3)=O)cc(O)cc(F)c1 CC(C)CCC(O)C(=O)N1CC(C(F)(F)F)CC1CNC(c1nc[nH]n1)=O C(=O)(C(C)(C)CCC#N)NCC12C(CN(C(C(C3CC(F)(F)C3)OC)=O)C1)CC2 C1(CNC(CC(C(C)C)O)=O)N(C(c2ccc3c(c2)CC3)=O)CCCC1(C)C N1(C(C2C(C)(C)CO2)=O)CCC(C)(C)C(NC(=O)CC2=NNC(=O)C2)C1 N1(C(Cc2nnc(C)o2)=O)CCC(CNC(c2cnc(C3CC3)o2)=O)C(C)C1 N1(CC(=O)N(CC(C)C)C2CC2)CCC(C(N(CC)CC)=O)CC1.c1cc(C)on1 S(=O)(=O)(c1ccc(C#N)c(NCCc2cc(F)ccc2Cl)c1)N(C(C)CS(C)=O)C N1(C(CCC=C)=O)CCCC(C(=O)NC2CC2CNS(=O)(=O)CCCOC)C1 N1(C(CCOC)=O)CCCCC1C(C)NC(=O)COc1ccc(F)cn1 N1(C(C2C(CCC)CN(C(=O)CCc3ccccc3)C2)=O)CC2CC(C)C2C1 c1(COC)c(C(=O)NC2CC2CNC(c2ccc(C(F)(F)F)nc2)=O)nnn1C c1(C2C(CNC(C(=O)NCC(CC)C)=O)C2)c(Cl)cccc1Cl CC(C)(C)CC(O)C(=O)NCc1cc(C(=O)NOCCc2ccccc2)no1 CC1=NN(C)C(=O)C1CC(N1CC(F)(F)CC1CCNC(c1nocc1C)=O)=O C1(C(N2CC3C(NC(c4c(OC)scc4)=O)(C3)C2)=O)CCCC(F)(F)CC1 C1(C(=O)NCCCN(C(=O)CCC2CC2(Cl)Cl)C)CCCCO1 c1(NCCCN(C(c2c(C)nc(CC)o2)=O)C)c([N+](=O)[O-])c(C)nn1C(C)C CC1CCn2cc(C(=O)NCC3(F)CC(NC(C4CCCNC4=O)=O)C3)nc2C1 C1(NC(COCCCCCC)=O)CN(C(=O)CCc2ccc(O)cc2)CC12CC2 C1(C(N2CCCC(Nc3ncc(Br)cn3)C2)=O)CCCC12CCOCC2 c1(C(=O)NCC2OCCN(C(CCNS(C)(=O)=O)=O)C2)cncc2cnccc12 c1(C(CC)NC(C)=O)nc(C2CC2(C)C)nn1-c1cnn(C)c1 C12(C(=O)Nc3ncn(C)n3)CCC1CN(Cc1sccc1Cl)C2 N1(C(Cn2c(C(=O)OC)cnc2)=O)C2CCC1C(NC(=O)CC(C)(C)C1CC1)C2 N1(C(C2(CCOC)CCC2)=O)CC2(C1)CN(C(=O)C=CC1(C)CCOCC1)C2 C(=O)(C1=CCc2ccccc21)N1CCC(O)(C(=O)NC(C)CC(C)(C)C)CC1 FCCCN=C(NCC1Cc2ccccc2C1)N1CCC2(CCCOC2)C1 N1(C(C2C(C)CC(=O)N2)=O)CCCC2CN(C(c3nnnn3C)C)CCC12 N1(CCC(=O)NCC(CCCC)NC(c2cc[nH]c2)=O)Cc2ccccc2C1=O c1(CN(C)C(=O)NC2(c3ccc(Br)cc3)CC2)ccc2c(c1)OCO2 CC1(C(=O)NC2CCN(C(c3cncc(Cl)c3Cl)=O)CC2F)CCNC(=O)C1 C1(C#N)(CC(=O)NCC(C(C)(C)C)NC(c2cnn(C)n2)=O)CCOCC1 N1(C(Cc2nc(C)oc2)=O)CCC(NC(c2ccn(C3CC3)n2)=O)C(C)C1 C1(C(N2C(C)(CCC)CC2)=O)C(O)CCN1C(C1CCC(=O)N1)=O CC1C(NC(=O)CSCc2cccs2)CCCN1c1cc(O)ncn1 c1(N(CC(C)C#N)C)ccc(S(=O)(=O)NCC2(C)CCCS2)cc1C#N CC1(C)CCC(C(N2CC(CC(F)F)C2)=O)(NC(=O)CN2CCNC2=O)C1 C(=O)(C1OC(=O)c2ccccc21)N1CC2CC(CN(C(C(C)O)=O)C2)C1 c1(C(=O)NCCCN(C)C(c2ccc(C(N)=O)cc2)=O)ccnc(Br)c1 CC1CCCn2ncc(C(=O)N(C3CN(C(C4CC5(CC5)C4)=O)CCC3C)C)c21 N1(C(C(CC)=CC)=O)C2CCC1CN(C(=O)C(C)NC(c1cccc(C)c1)=O)C2 C1(C)(C(=O)NC(C(=O)NC(c2nc[nH]n2)CC)CO)CCN(C)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N(C(CCNC(c1c(C)nn[nH]1)=O)C(C)C)C C1(CC(=O)NCC(CC)(C)CC)CC(C)(C)CN1C(=O)CC(C)(C)OC C12(NC(c3c(Cl)cc(C)c(C)c3)=O)COCCC1CN(C(c1cccnn1)=O)C2 c1(C(=O)NC(C2CCN(C(c3ccc(O)nc3Cl)=O)CC2)C)cncn(C)c1=O C#Cc1ccc(Cl)c(C(N2CC3(CCN(C(=O)CC4CC4C)C3)C2)=O)c1 Cc1cc(CC(C)C)nc(NC2CC2CC2CC2c2ccccc2Br)n1 CCCCCC(O)CC(=O)N1CCC(CNC(=O)C(C)CC2CCCC2)CC1 CCCCCCCCC(F)C(=O)NCC1(CO)CCN(C(=O)C(O)C(F)(F)F)C1 N1(S(CCOC)(=O)=O)CCN(C(=O)CCc2cnn(-c3ccncc3)c2)CC1 c1(OC)c(C(N2CCC(NC(=O)C=CC(F)(F)F)CC2)=O)c(C)nn1C C=C1CCC(C(N2CCC(CN(C(=O)CCCCC3CCCCC3)C)C2)=O)CC1 CC(C)CCCC(=O)N1CCC12CN(C(=O)CC1(O)CCC1)C2 c1(C(N(CCC(=O)NC(c2nnnn2C2CC2)C)C2CC2)=O)ccc2c(c1)CCC2 S(=O)(=O)(c1nc(N2CCOC(C3CC3)C2)ccc1Br)NCC1(CC)CCCO1 N1(CCNC(CN2CCN(C)CC2)=O)CC(=O)Nc2ccccc21 c1(COC)nc(C(=O)N(C(C)CCNC(=O)CCc2nccn2C)C)co1 c1(CC=C)cc(C)ccc1C.n12nc(-c3ccc(Cl)nc3)nc1c1ccc2cc1 C12(C)CCN(CC1)C2=O.c1cccc(O)n1.C(CC(F)=C(F)F)c1cn(CC)nn1 C(=O)(C(C(=O)NCC(O)CNC(c1cc2cnn(C)c2s1)=O)C(C)(C)C)OCC CCCC(O)C(=O)NCCCCCN(C)C(C1COC(C)(C)C1)=O Cc1c(F)ccc(CN2CC(C)(C(=O)NC(CO)C(C)O)C2)c1Cl N1(C(CCC#CC)=O)CCC2CCCN(C(c3c(Cl)sc(C)c3C)=O)C2C1 c1(C(=O)NCC2N(C)CCN(C(C(CCC(C)C)O)=O)C2)c[nH]c(=O)c2ccnn12 N1(C(CCc2cn(C)nc2)=O)CC2(CC(C(=O)NC(C)(C)COC(C)C)CO2)C1 CCC(CC(=O)NCCC1CC(NC(=O)Cn2ccnc2)C1)C1CC1 C(=O)(CCC(C)S(C)(=O)=O)N(C1CCN(C(=O)CNC=O)CC1)CCC N1(C(C2(C#C)CCN(C(=O)CCOC3CCC3)C2)=O)CC2CCCC(C1)N2C CC(C)C(C#N)C(=O)NCc1nnn(C)c1C(=O)NCC1CCCOC1 C1(CC(=O)NC)CN(C(=O)CCS(C)=O)CCN1C(C1CC=CC1)=O c1(C(=O)NCC2CCN(C(CC(=O)NC)=O)C23CCC3)ccc2c(c1)ncn2C c1(CS(N2CCN(CC(=O)N(C)C)CC2)(=O)=O)cccc(C#N)c1 c1(C(=O)NCC2CN(C(CC3CC(OC)C3)=O)CC2(C)C)cn2ccnc2cn1 C(CCCCCNC(=O)CN(C)CCO)N(C(c1c(C)n[nH]c1)=O)C CCCCC(C(=O)NC1CC2(C1)CC2NC(C1CC(C)C1)=O)NC(N)=O C1(CC(=O)NCC2CCN(C(c3scc(C)c3)=O)C2(C)C)CC2(CCCC2)CO1 CC1CN(C(=O)C(c2ccn(C)n2)N)CCS1(=O)=O N1(C(CC2=NNC(=O)C2)=O)CC(C2CCCCN(C(c3scnc3Cl)=O)C2)C1 C(=O)(C#CC(C)(C)CNC(=O)C(C)(C1CC1)OC)N1CC(C(=O)NC)C1 C1(CNC(Cc2c(C)n[nH]c2)=O)CCCCC1NC(c1cnn(C)c1F)=O C#Cc1cccc(CNC(=O)CCCN(C(=O)COC)C(C)C)c1.C1CC1 C1(C(N(C2CCCC2)CCNC(CC(=O)OC)=O)=O)CCn2cc(C)nc2C1 C(c1ccccc1C#N)=CC(=O)NC(CCNC(C(CSC)C)=O)C(C)C C(=O)(C1=C(Cl)CC1)N(C1(CO)CCC1)C1CC1.C12(OC)CN(C1)C2=O c1(C(N2C(CNC(C3CN(C)C(=O)N3)=O)COCC2)=O)coc2c(Cl)cccc12 CC1CN(C(=O)CNC(=O)C(C)(C)C)CCC1NC(=O)Cn1cnc(C#N)n1 C1(CNC(C(c2ccc(Cl)cc2)(C)C)=O)CN(C(C2(C)CC2(F)F)=O)CCO1 N1(c2cc(C)nc(C)n2)CC2CCC1C1CN(C(=O)Cc3ccccc3F)CC21 c1(CC)ncc(C(=O)NCC(C)(C)CC2CN(C(=O)C(C)N3CCC3)C2)c(O)n1 C1(CNC(=O)CC2(O)CCCCC2)CN(C(=O)Cc2ccnc(F)c2)CCCO1 CC(C)CC(C)CC(=O)NCCn1cc(C(=O)NC(C)CCC(C)(C)C)nn1 c1(C(N2CC(N(C(C(C)n3cnnn3)=O)C)C2)=O)ccnc(N2CCC(C)C2)c1 N1(C(CNC(=O)NC)=O)C2CCCC1CN(C(=O)CC1(C#N)CCOCC1)CC2 C(CC(O)C(=O)NCC1(c2ccon2)CC1)NC(C1C(C)C1C)=O c1(CC(=O)NC2CCN(C(=O)C(c3ccccc3Cl)O)C2)cccc(C(F)(F)F)n1 O=C(C1=NOCC1)N1CCC(c2nc[nH]n2)CC1.c12nocc1NC2=O C1(CNC(CN(S(C)(=O)=O)C)=O)(CO)CCN(C(C2OCCC2C)=O)CC1 C1(CNC(C=CC)=O)CCCC1NC(=O)C(F)Cc1ccccc1 n1(CC(=O)N(C2C(C)CCN(C(C3(CF)CCC3)=O)C2)C)cnc2ccccc12 CC1(C#CC(=O)N2CCCCC2CNC(C2CCC3CCC23)=O)CC1 N1(CC)CCCC(C(N2CCC2CNC(=O)C=Cc2ccc(C(N)=O)o2)=O)C1 c1(NC(=O)Nc2cc(C)c(NC(C3CCCCC3)=O)cc2)ccn2nnnc2c1 N1(C(c2c(Cl)cn(C)n2)=O)CCCN(C(C2(O)CC2)=O)CC1 Cc1[nH]nc2ccc(C(=O)N(C)CCOCCCN(C)C(c3cc[nH]c3)=O)cc12 c1(NC(C2CC23CN(C(C2COCCO2)=O)C3)=O)c[nH]ccc1=O C1(c2cccnn2)(NCC(C)(C)CC=C(C)C)CCC(P(C)(C)=O)C1 c1(SC)cn(C)nc1C(=O)NC(C)CC1CCN(C(=O)CC(F)(F)F)CC1 c1(C(N2CCC(CN(C)C(c3nn(C)cc3N)=O)C2)=O)ccc2nn[nH]c2n1 CC1(C)CCC(CNC(C2CC2[N+](=O)[O-])=O)N(C(c2cnc(S)nc2)=O)C1 C(CCC(=O)NCC(CNC(c1cnn[nH]1)=O)CO)NC(=O)OCC C(c1ccccc1)=CC(=O)NC(C1CCCCC1)CO c1(NC(c2cn(CCN(C)C)nc2)=O)ccccc1C1CCCCC1 c1(OC)c(Br)ccc(CNCC2CCCN(c3cc4ncnn4cn3)C2)c1F C#Cc1ccc(C(N2CC(NC(=O)CC3CCCC3O)C(F)C2)=O)cc1 C1(C2CCC2)(C(=O)NCC(CNC(c2csc(C(C)C)n2)=O)OC)CCC1 c1(C(=O)NCC(CNC(C(C)(c2cccs2)N(C)C)=O)(C)O)ccc(F)cc1F N1(C(C(C(C)C)N(CC)CC)=O)CCC(C)C(CNC(=O)CC2=CCCC2)C1 c1(NS(C)(=O)=O)ccc(NC(=O)NC2CN(C(=O)CN3CCNCC3)C2)nc1 Cc1cc(C(N2CC(F)CC2CNC(=O)C(C)(C)Cc2cnn[nH]2)=O)ccn1 c1(OC)cccc(C2(C(=O)NCC3CC3NC(=O)CC3CCCC3)CC2)c1 N1(C(c2cn(CC(C)O)c(=O)cc2)=O)CC(NC(=O)CCC2CC2)C(C2CC2)C1 C1(C(=O)NC(CN(C(C(COC)C)=O)C2CCCC2)C)C(C(F)(F)F)C1[N+](=O)[O-] c1(CCC(=O)NCC(C)(C)NC(CC(C)SC)=O)cc(F)c(F)c(F)c1 N1(C(C2CCC(C)CC2)=O)CCC(CNC(=O)CCc2cccs2)C(O)C1 c1(C2(C(=O)NCCCN(C(=O)CCCF)C(C)C)CCC2)ccc(Br)cn1 C1(N(C(CCNC(C)=O)=O)C)CN(C(C2CC(N3CCOCC3)C2)=O)CC1F N1(C(C2N(C(C(C=C)(F)F)=O)CC3CCCC32)=O)CC2CCC1C(O)C2O Cc1cnc(C(N2CCN(C(C3CC(=O)N(c4ccccn4)C3)=O)CC2)=O)cn1 C1(NC(C(CC)N2CCCC2=O)=O)CC(NC(=O)C(C)=C(C)C)C(O)C1 c1(C(=O)NCC2(CC(=O)N(C)CCc3ccccc3)CC2)ncn2c1CCC2 c1(OC)cc(NC(c2ccc(Cl)cc2F)c2nnnn2C(C)(C)C)cnc1OC N1(C(C(C(C)C)NC(=O)OC)=O)CCCC(C2CN(S(=O)(=O)CC#N)C2)C1 N1(C(c2cc(C)oc2)=O)CCCC(CCNC(=O)CC23CCCC2C3)CC1 C1(NC(CCn2ccc(C)n2)=O)CN(C(=O)CCCCC(C)C)C2CCCC12 C1(NC(CSCCC)=O)CN(C(=O)CCOC)CCC1c1ccc(F)c(F)c1 c1(N2CCN(C(C(CC)CO)=O)CC2)cc(Cl)ccc1OC(=O)OCC N1(C(C=C(CCC)C)=O)CC2(CCCCN2C(c2cc(C)co2)=O)C1 C1(CNC(Cc2cc(C)nn2C)=O)CN(C(C2CCC(=O)N2C)=O)CC(C)(C)C1 C1(CCNC(=O)CC2CCCC2)CN(C(c2ccsc2Cl)=O)CCCO1 C#Cc1ccc(NCc2ccccc2)nc1.C1(C(F)F)CC(=O)Oc2cccc1c2 CC1(C)CCCC(CC(N2CCC(OCC(N3Cc4c[nH]nc4C3)=O)C2)=O)O1 c1(C(=O)NCC2(CNC(C3CCCS3)=O)CCCC2)n[nH]c2ccc(O)cc12 C1(CC(=O)NCCN(C(C)C)CC)CC(O)CN1C(=O)CCc1ccc[nH]1 c1(C(=O)NC)ncnc(O)c1F.c1(CC)ncoc1C(=O)N(C)CC1(CCO)CC1 c1(C(C)C)ccsc1C(=O)NCC1COCC1NC(C1COCCO1)=O C1(C(=O)NCC2C(CNC(c3ccc4nn[nH]c4n3)=O)C2)CCc2nn[nH]c2C1 C1(C)(C(=O)NC(C)CF)CCCN(C(c2c(Cl)cccc2I)=O)C1 C1(NC(CCCn2c(C)cc(C)n2)=O)CCN(C(c2n[nH]cc2F)=O)C(C)C1 CCC(C)(C#N)C(=O)NCC1CN(C(=O)CC2CCC(C)CC2)CCO1 CC1CCOc2c(C(=O)NCCCOCCO)cccc21 C1(CCNC(c2ccc(F)s2)=O)CC(F)(F)CN1C(=O)COc1ccc(O)cc1 Cc1c(C(=O)NCC2CC(NC(=O)CCC(C)N(C)C)C2)[nH]c2cc(F)ccc12 Cc1cccc(OCC(N2CCC(C3CCCN3C(=O)CC(C)(C)C)C2)=O)c1C S(=O)(=O)(c1ccc(OC)c(Cl)c1)N1C2CN(c3nc(SC)nc(C)c3Br)CC21 C1(NC(c2cn3ncnc3nc2C)c2n(CC)nnn2)Cc2ccccc2C1 C1(C(=O)NCC(CNC(CC2CC(SC)C2)=O)CO)C2(CC2)C12CC2 c1(C(=O)NCCN(CCOC)C(C2CC3C=CC2O3)=O)cn2ccc(C)cc2n1 c1(C(N2CCN(C(C(CC#C)(C)C)=O)CC2)=O)cc[nH]c(=NC)c1[N+](=O)[O-] CC(C)CCC(F)C(=O)N(CC(N1CC(CO)C(C)(C)C1)=O)C Cc1oc2cc(C(=O)NCC3CCCN(C(C4(CO)CCCO4)=O)C3)[nH]c2c1C C1(N(C(CSCC(=O)OC)=O)CC2CCCO2)CCN(C(c2ccsc2)=O)C1 C1(CC(C)NC(c2scc(COC)c2)=O)CCN(C(C2(C#N)CC=CC2)=O)CC1 N1(C(C(CNC(c2cn(C)c(=O)cn2)=O)OC)=O)CC(C2=NOC(C)C2)C1 N1(C(C(C)CC(F)F)=O)CCN(C(=O)C(C)(C)COC2CCCC2)C2(CC2)C1 c1(CN(C(=O)C(C)CN(C(=O)CCCF)C)CC)ccccn1 N1(C(CCCCC)=O)CC(C(=O)NCc2ccccc2CC)C2(CC2)C1 Cc1coc2ccc(C(=O)NC3CC(CNC(=O)C(F)(F)C(F)(F)CO)C3)cc12 c1(C(N(C2CC2)CC2CCN(C(C=CC)=O)CC2)=O)cnc2n1CCCCC2 N1(C(CCCOC)=O)CCC2CC2(C(=O)NCc2nncs2)CC1 C1(CNC(CNC(=O)NC)=O)CCN(C(=O)CNC(C)=O)CC1C C1(NC(c2cccc(C(N)=O)c2)=O)CN(C(=O)Cc2csnn2)CC12CC2 CCCCCCCC(=O)NC1CC(NC(c2cnn(CCC#N)c2)=O)C1 c1(NC(c2ccncc2)=O)ccccc1OCC1(C)CC(C)C1 c1(C(=O)NC2C=CCN(C(C3CCCCO3)=O)C2)c[nH]c2nc(F)ccc12 Cc1ccc2c(c1)CN(C(C1CC3(CCN(C(C4CCCCC4F)=O)C3)C1)=O)C2 C1(NC(C(C)C)=O)CC(O)CN(C(C2CCC(C#N)CC2)=O)C1 c1(C(=O)OC(C(=O)OC)c2ccoc2)cc(C(C)=O)cs1 c1(C(=O)NCC(C(C)C)N2CCCCC2)cc(C(F)(F)F)nn1C C1(NC(C2(OC)CCSC2)=O)CN(C(=O)Cc2cc(C)cc(CO)n2)CC1(C)C c1(C(=O)NC2CCC(NC(=O)COCC(F)F)CC2)cc2n(n1)CCCNC2=O N1(C(c2c(C)noc2C)=O)CCCC(NC(=O)COC2CCCCC2)CCC1 C(C#Cc1cn(C2CC(O)C2)nn1)NC(=O)CCC1CCCC1(F)F C(=O)(C(CC)C(=O)NCCOCC(=O)N(C1CC1)Cc1cccs1)OC C(=O)(C(Cc1cc[nH]n1)NC(=O)OC(C)(C)C)N1C(CC)CC1 C=CC1(C(=O)Nc2cccc(C)c2)CCN(C(=O)C(F)CC(C)(C)C)CC1 C1(C(N(CCNC(Cn2c(C(=O)OC)ccn2)=O)CC2CC2)=O)C2(CC2)C12CC2 c1(C(N2CC(CNC(CCSC)=O)CC2(C)CO)=O)nccc2ccccc12 C1(C(N2CC3C(CC(NOCC(=O)OCC)=O)(CC3)C2)=O)CCCCC(=O)CC1 c1(C(=O)NC(C(C)C)CNC(C2(C)CCC(C)C2)=O)ccc2c(c1)C(=O)NC2 C#Cc1cc(NC(C2CN(C(=O)Cc3ccc(F)cc3)CCO2)=O)ccc1C C=CCCCCCNC(=O)C(Cn1cncn1)NC(=O)CCCC#N N1(C(CCCC=C)=O)CCCC1C1CCCN1C(c1ccc(C#N)c(O)c1)=O C1(C(N(C2CCN(C(=O)OC(C)(C)C)C2)CC)=O)CCCN1C(C)C C1(N(C)C)CN(C(CCCc2cccc(OC)c2)C(=O)OCC(F)F)CC1(C)C c1(C(=O)NCCC(C)NC(=O)C=CC2CCCO2)ccc2nnn(O)c2c1 CCC1=NOC(C(=O)N(CCC(=O)N(CCCO)CC(C2CCCO2)O)CCO)C1 Cc1cc(F)c(C(=O)NC(CNC(c2cnc(-c3cccs3)o2)=O)CO)c(Cl)c1 C(=O)(CC(C)C(=O)OCC)N1C(C(=O)NC2CCN(C(CC)=O)C2)C=CC1 C#Cc1cnc(C(N2CCC(N(C)C(C34COCC3C4(F)F)=O)C2)=O)c(C)c1 C(=O)(C1CCCc2c[nH]nc21)NCCC1(NC(C(CCC)C)=O)CCC1 N1(C(C2CCC2NC(C23CC(F)(C2)C3)=O)=O)CCCC2(C=CCO2)C1 CC(C)(C#N)CCC(=O)N1CC(OC(=O)C(C2(S(C)(=O)=O)CC2)c2ncccn2)C1 C#Cc1ccc(C(N2CC3(NC(C4COCCN4C)=O)CCC2C3)=O)cc1 CCCCCCC(C)(C)C(=O)NC1CC(CNC(=O)C#CC(C)C)C(O)C1 C(=O)(C(C)CCC(C)(C)C)N(CCCCC(=O)NCc1cc(C)sc1)C c1(CN(C(c2cnn(C)c2)C(=O)NCC2CC2)CCC)cccnc1.C(CC)S C(c1ccco1)=CC(=O)NC(C(=O)NCCC(=O)NC(N)=O)C1(O)CCC1 c1(C(=O)OCC)coc2ccc(NC(C3(C)CCCN(CC)C3)=O)cc12 N1(C(COC(CC)CC)=O)CCCC(NC(C2CC2C(C)(F)F)=O)C1C c1(C(CC2CCC2)NC(CC(C)c2ccccc2)=O)ccc(Cl)cc1 N1(C(=O)NC(CCC)(C)C)CCCC(CN(CC)CC)C1 C(=O)(C(F)(F)C(F)F)NCC(CC(=O)Nc1cnn(C(C)(C)C)c1)OC C12(C(=O)OCN)C3C4C1C1C2C3C41C.C12(O)CCN(CC1)C(=O)CC(=O)N2 C(=O)(CC(F)(F)Cl)NCCC(=C)CNC(=O)C(c1ccc(OC(F)(F)F)cc1)C C1(CNC(C2C(C)(C)C2(C)C)=O)C(C2CC2)CCN1C(=O)CCC(CF)CF C12(C(N3CC(NC(c4n(C=C)ncc4)=O)C(F)C3)=O)CCCCCC1OCC2 C1(CC(=O)NC(CNC(C(C2CCCCC2)C)=O)CO)C=NN(C)C1=O C1(C(=O)NCC2(C(=O)NCC3CCOC3C(C)C)CC(=C)C2)CCCSC1C C1(C(=O)NCC2CC(F)(CNC(C=C3CCC(C)C3)=O)C2)CCCCN(C)C1=O C(=O)(C1=C(C2CCOC2)N(C2CC2)C(=O)NC1c1nc(Br)cs1)OC N1(C(c2c(C)cc(C#N)cc2)=O)CCC2OCCN(C(C3CCCOC3)=O)C2C1 c1(C(N2C(C(=O)NC(CC)C(C)CN(C)C)(CC)CCC2)=O)cncn(C)c1=O N1(C(C(C)C#N)=O)CCCC(N(C(=O)CCOc2cccnc2)C)C1 C1(n2cc(C(=O)OC)nn2)CC2CCC1(NC(c1cccc(Cl)c1F)C1CC1)C2 c1(CNC(C2(n3cc(C(CC)O)nn3)CC2)=O)cc(C)c(F)cc1Cl C(=O)(C(C)(C)CF)NC1C(NC(C=COC(C)C)=O)COC1.c1(C(C)OC)ccccc1 c1(OC)cc(C(=O)NCC(C)NC(c2n[nH]c(C3CC3)c2Cl)=O)cc(Cl)c1 C1(NC(Cc2ccc(C)cc2)=O)CN(C(c2ccon2)=O)Cc2ccnn2C1 C1(=CC(=O)NCCN(C(C(C)n2ccnc2)=O)C)C2CC3CC(C2)CC1C3 Cc1cc(O)c(C(N2CCC(NC(C3CC(C)CO3)=O)C2(C)C)=O)nn1 C1(NC(C2CC(C)CN2C(=O)CC2CCC(=O)N2)=O)CC(C)(C)C12CC2 c1(CN=c2ccn(CC(N3CC4CC(C3)O4)=O)c(O)n2)nccc2ccccc12 c1(OCC)ccc2ccc(-c3cc(C(=O)NC(=O)NC(C)C)ccn3)cc2n1 C1(CC)CC(C(=O)NC(C=CC(N2CCC(CC#C)C2)=O)C)CCO1 N1(C(CN(C)C(C2CC3CCC2O3)=O)=O)CCN(C(=O)C(F)CC2CCC2)CC1 C(CN(CC1CC=CCC1)N(C)Cc1cnn(C)c1)OC N1(C(c2scc(OC)c2)=O)CCCC(C(=O)NCCN2CCC2)C1C N1(C(C2CN(CC)C(=O)CC2)=O)CCC(C)N(C(=O)C(O)C2CCC2)CC1 [N-]=[N+]=NCCCCC(=O)NCC1CCCC1NC(c1ccc(C(F)(F)F)[nH]1)=O CON1CCC(CC(=O)NC(CO)C(C)NC(c2cc(CN(C)C)on2)=O)CC1 c1(CC)nc(C)c(C(=O)NCCC2CCCN2C(=O)CCc2ccnn2C)s1 c1(C(N2C(C)(C(=O)NC(C(C)F)C)CCC2)=O)ncn2ccccc12 c1(NC)ncccc1C(=O)NCC(C1CCOC1)NC(=O)CC(C)(C)OC C(=O)(C(C)(O)CC(C)C)N1CCN(C(CC2C(C)=NNC2=O)=O)CC1.C1C(=O)N1 c1(OC)cc(CNC(=O)CSC(C)(C)C)ccc1OC(=O)C(C)OC c1(C(N2CC(NC(C3C4COCC34)=O)C(F)CC2)=O)cccc2nc[nH]c12 Cc1ccn(CC(C)C(=O)N(CCCCNC(c2scnc2C)=O)C)n1 C1(NC(c2nccc(OC)c2F)=O)CN(C(=O)CC2(CO)CCC2)CC12CCC2 CN(C)S(=O)(=O)N(C)CC(=O)NCCC(C)(C)NC(c1cc2[nH]ccc2s1)=O C1(CC(=O)N(C(C(=O)OC)C)C)CCCCC1NC(=O)CC1CCC(O)C1 CC(C)C(C(=O)NCC(C1CCCCC1)NC(=O)CCCC#N)NC(N)=O C(CCCC(=O)NC(C1CCCC1)CNC(C1(Cl)CC1C(C)=O)=O)N(C(C)=O)C C1(C)(C(=O)NC(CCCNC(CSCC=C)=O)C)CCCS1 C(CNC(=O)CN1CCC(N(C)C)CC1)(CC(F)(F)F)NC(C1(CC=C)CC1)=O N1(C(C(C)N(CC)CC)=O)CCC2(CCCN2C(c2coc(C(F)F)n2)=O)CC1 c1(C(N2CCC(CCC(=O)NCc3ncn(C)c3)C2)=O)ccsc1C#N N1(C(COCCCCCC)=O)CCC(C(=O)N(C)CCc2cccs2)CC1 CCC(C)CCCC(=O)NCC1(C)CCCN1C(c1cc(CO)oc1C)=O CCC1=C(C(=O)NC2CCCC2NC(C2(C#N)CCCO2)=O)SCCO1 CCS(=O)CC(=O)NCC1CN(C(c2ccnc(F)c2)=O)C1 CC1(C)C(NC(C2(CNC(C3CCCN3C3CC3)=O)CC=CC2)=O)CC1(F)F N1(C(c2c(C)ncn2O)=O)CCC(NC(c2ccsc2Cl)=O)C(F)(F)CC1 n1(CC(N2CCN(C(C(CC)C)=O)CC2COC)=O)cc([N+](=O)[O-])c(C)n1 c1(NC(c2cc(C)c(Br)cc2F)=O)ccc2c(c1)CN(Cc1cccnc1)C2 Cc1cc(Br)ccc1CCC(=O)NC1CCN(C(c2ccc(F)s2)=O)C1 c1(C(=O)NC2C(CNC(=O)CSCc3ccccc3Cl)C2)cc2cccn2cn1 N1(C(C(CC#C)C2CC2)=O)CCC2C(C1)CN2C(=O)Cc1csc(CC)n1 Cc1ccc(C(=O)OC2CCC2)c(C)c1.N12CCCCC1C(=O)NCC2=O.C(CO)O C(C(C(=O)NCCn1cc(CO)nn1)NC(=O)C(O)CC1CCCC1)SC c1(C(N(C)CC=CC(=O)NCCc2cnn(C)c2)=O)cc(C)sc1C N1(C(C2(C(=O)OCC)CC2)=O)CCN(C)CC1CC.c1(C(=O)NC)cn(C2CC2)nn1 C1(OC)CCCC1C(N1CCCC1Cn1cc(CNC(C2CCCS2)=O)nn1)=O CC1CN(C(C2C(CNC(c3cnsn3)=O)C2(C)C)=O)CC(C)(C)C1 C(CC(C)(C)CC(=O)NCCC1(NC(C2SCC=C2C)=O)CCCC1)OC CCCS(=O)(=O)NC(C)C(=O)NC1CC(NC(=O)CC2(COC)CC2)C1 c1(C(=O)NC(C(C)NC(C(C(CC)O)C)=O)C)cnc2ncnn2c1O C1(NC(C2CCC(O)CC2)=O)CC2CCC(C1)N2C(c1ccns1)=O c1(C(=O)NC2CC2CNC(C2(C3CCCCO3)CC2)=O)cncc2ccccc12 C=C(Cl)CCC(=O)NCCCOCCNC(c1cc(-c2ccccc2Cl)[nH]n1)=O C1(CNC(C2(COC)CC=CC2)=O)C(C)CCCN1C(=O)CCC1CC1(C)C CCC(C)C(CC(=O)NC1CN(C)C(C)(C)C1)NC(=O)C(C)(CO)OC S(=O)(=O)(CC(=O)NCCCN(C(C1(C)CCCOC1)=O)C1CC1)N(C)C N#CC1(C(N2CCC(O)(CNC(=O)Cc3ccco3)C2)=O)CC2CCC1CC2 c1(C(N(CC(C)N(C(c2nn(CC)c(O)c2)=O)C)C)=O)ccc2c(c1)COCO2 c1(C2C(C(=O)Nc3ccc(CNC(C(C)CF)=O)cn3)C2)cccc(C#N)c1 c1(N2CCC(O)(CC#N)CC2)nc2ccc(Cl)cc2c(=NC2CCCCCC2C)[nH]1 c1(C(N2CCC(NC(CC=C=C)=O)CC2C2CC2)=O)cncc2c[nH]nc12 C#CCCC(C(=O)NC(COCC)CO)NC(C1CCN(C)C1CC)=O C12(CC)CN(C(=O)C(c3cccc(C)c3)F)C(CNC(C3CN(C)C3)=O)(C1)C2 C1(NC(C2CCC(C)N(C(=O)COC3CC=CC3)C2)=O)CCCC(F)(F)CC1 C(=O)(CCC(F)F)N(C1CCN(C(=O)C(c2ccc(Cl)cc2)CO)C1)C c1(C(=O)NCC2C3CN(C(=O)CC4OCCCO4)CC23)occ2c1CCC2 N1(C(C(=Cc2cc[nH]n2)C)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1CCO c1(OC)nc(C(N2CC3CCC2C3NC(=O)C(F)C(C)C)=O)cc(O)n1 C1(OC)(CNC(C2(C)CCSCC2)=O)CCN(C(=O)Cn2nc(C)nc2C)C1 CC1CC2(CC(C(N3CC(O)CCC3C(=O)NCC3CC(C)(C)C3)=O)C2)C1 N1(C(C2(COCC)CC2)=O)CC2(CC(NC(=O)C(c3cccc(C)c3)C)C2)C1 C(CCCCCNC(=O)C(c1ccc(F)cc1)O)NC(=O)CC(F)F N1(C(c2c(C)coc2)=O)CCN(C(=O)COC(F)F)CCC1C C1(C)(C(=O)OCC)CCN1Cc1cnc(C2CCCO2)s1 c1(CC)nc(C)c(CC(N2CCC(C)(CNC(=O)C(C)CC)CC2)=O)c(C)n1 C1(CC=C)(C(C)C)CN(C(c2cn(C)nn2)C(=O)NCCC2(C)CC2)CCO1 c1(OCC=C)ccc(CC(=O)NCCC(O)CNC(c2ccc(OC)s2)=O)cc1 C=CCC(C)C(=O)NCC1CCC1NC(c1oc(-c2cnn(C)c2)nc1C)=O c1(CC)noc(CCC(=O)NC(C)(CNC(c2cc(COC)c[nH]2)=O)CO)n1 C1(CNC(C(F)=C(C)C)=O)CN(C(c2csc(C)c2N)=O)CCC12CCC2 c1(C(N2CC(NC(CN3CC(C)C3)=O)C(F)C2)=O)cccc([N+](=O)[O-])c1Br c1(C(C=CC=CCC)C(=O)OC(=O)C(C)C)ccccc1 C(N=c1[nH]c2cc(F)ccc2s1)c1[nH]cc(S(=O)(=O)NC)c1 C(=O)(CCCC(=O)NC1(CN)CN(c2nncs2)C1)C(c1cccnc1Cl)=O C1(NC(CC=C=C)=O)CCN(C(C2CC(C3CCC3)C2)=O)CC1(C)C C1(F)(C(=O)NCC2CCN(C(C(C)Oc3ccc(Cl)cc3)=O)C2)CCOCC1 C=CC1CN(C(=O)C(C)P(C)(C)=O)CC1NC(=O)CC(C)(C)COC C(=O)(CCCCCCN(C(=O)C(O)CN(C)C)C1CC1)Nc1c(C)cc(O)cc1 N1(C(CSc2c(C)[nH]c3ccccc32)=O)CC(CN)CC1C1CCCC1 C1(NC(c2nn(C)c(Cl)c2)=O)CCC2(C1)CN(C(C1CCC(O)CC1)=O)C2 C1(F)(CNC(c2cccc(F)c2Cl)=O)CCCN(C(c2cscn2)=O)C1 C1(NC(CC(C(C)C)C)=O)CCN(C(c2cnc(C3CC3)o2)=O)C12CCCC2 c1(OC)n[nH]cc1C(=O)NCC1CC1C(=O)NC(CO)CCF C1(COC)CN(C(=O)C(CCSC)N2CCC(OCc3ccccc3)C2)CCO1 c1(OC(C)(C)CNC(=O)C(c2ccoc2)NC(C2CC(C#N)C2)=O)cccnc1 c1(CCC)nc(C(=O)NCC(C)CN(C(=O)C(C)c2cncs2)C)co1 C1(C(=O)NCC(O)COC)(CNC(CNC(CC)=O)=O)CCCCC1 C#Cc1ccc(C(=O)N(C(CC)C(=O)N(C)CC2(O)CCCC2)C)o1 Cn1cnc2ccc(C(=O)NCC3CN(C(=O)C(N)=O)CCO3)cc12 c1(C(CNC(C(C)(C)OC)=O)NC(c2ccc(CO)s2)=O)cccc(C)c1 C(=O)(CC1C(=O)N(C)c2ccccc21)NCC1=CCN(C(C2(C)C(C)C2)=O)CC1 c1(C2N3CCN(CC3)C(C#C)CNC2=O)ccc2c(c1)CN(C)C2=O.C1(CC)CC1 Cc1nnccc1C(=O)NC1CCCC1CNC(=O)C(C)(C)c1cnco1 CS(=O)(=O)CC(=O)NC12CC(CNC(=O)CCNC(c3ccc[nH]3)=O)(C1)C2 N#CC1CN(C(c2cccc(Cc3cn(C4CC(O)C4)nn3)c2)=O)CC12CCC2 c1(CC(N2CC(C)C(NC(=O)CC3CCCC34CC4)C2)=O)c(O)ncnc1O N1(C(C(=O)NC(CC)(C)C)c2cn[nH]c2)CCOC2(CCC(C)(C)C2)C1 N1(C(=O)Nc2nc(COC)sc2)CC2CN(Cc3ccccc3)CC2C1 C(=O)(C1=C(C)OCCS1)N(C1CCCN(C(C2CSCN2C(C)=O)=O)C1)CC c1(C(=O)NCC2(NC(c3c(O)ccc(C)n3)=O)CCOC2)cc2n(c1)CCCC2 C1(CCCNC(c2cscn2)=O)COCCN1C(=O)C(C1(O)CCCC1)F N1(C(c2cnc(CC)[nH]2)=O)CCC(CNC(c2cc(C)on2)=O)(OC)C1 C1(CNC(CC(=C)C)=O)CN(C(=O)C(c2cnn(C(C)(C)C)c2)=O)CC12CC2 CC(C)(C(=O)N1CC(CNC(=O)CNc2ccccc2)C1)C(F)(F)F C1(C(C)NC(C2CCOCC2)=O)CCN(C(c2cnc(C(C)(C)CF)o2)=O)CC1 CC(=O)CCC(=O)N(CC(=O)NCCC1OCCC1(C)C)C(C)C C=CCCCCC(C(=O)NC1COC1)N1CCCC(C(CC)CC(CC)SC)C1 C(=O)(C1CCCn2nccc21)N1C(CNC(C2N(CC)CCC2)=O)CC1 N1(C(CSCCCC)=O)CC=CC(C(N2C(CO)CC2C)=O)C1 N1(C(C(=C)F)=O)CCC2CN(Cc3c(OC)ccc(F)c3Br)CC12 c1(-c2cc(C(=O)NCCCN(C(=O)C(CO)OC)CC)on2)ccc(Cl)cc1 C1(C2(O)CN(C(c3cccc(OCCF)c3)=O)C2)(CNC(C(C)O)=O)CC1 CC(C)C1=CCC(NC(=O)CCC2CCCN2C(C23CCN(CC2)CC3)=O)CC1 N1(C(c2ncn(CC)c2)=O)CC(NC(c2cc(C(N)=O)co2)=O)C2(CC2)C1 N1(C(C)=O)CCC(NC(c2cnns2)=O)C(CO)C1.[nH]1cc(C(C)(C)C)nn1 c1(C(C)=O)cc(C(=O)NCC2(CNC(=O)CCNC(N)=O)CCC2)cnc1C C1(NC(C(C(C)C)c2cnn(C)c2)=O)CC2CCC1CN2C(c1cncn1C)=O C1(C(N(C2(CC(N3CC(c4ccon4)C3)=O)CC2)C)=O)CCC(=O)NC1 N1(C(C2(CC=C)COC2)=O)CC(NC(c2coc(C3CC3)n2)=O)CC(C)C1 c1(CC(=O)NCCOC)cccnc1Cl.N12CC(CCO)(C1)NCC2=O.C(CN)OO c1(C(=O)NC(C)CCNC(=O)C(C(C)O)N(C)C)ccc2cncc(Br)c2c1 CC(CC(C)(C)C)C(=O)N1CCN(C(c2ccnc(C3CC3)c2)=O)CC1CO C#CC1CCCN(C(C2CCN(C(=O)OC(C)(C)C)C2COC)=O)C1 c1(C(N2C(C(=O)O)CCC2)=O)ccccc1Cl.C(C(Cl)C(=O)N1CCCC1CO)OC C(C(C(=O)NC1CCN(C(c2ncoc2-c2cnn(C)c2)=O)C1)N(C)C)OC Cc1ccc(CNc2cncc(NC(=O)C(O)C(C)(C)C)c2)c(Br)c1 c1(C(N2CC3(CN(C(CC(C(C)C)C)=O)C3)C2)=O)nc(Cl)cc(N)c1Cl N1(C(CCSCC#C)=O)CCC(CNC(c2cccc(NC)n2)=O)CC1C c1(Cc2ncc(NCCC3CCCC3)cn2)cc(Cl)ccc1Cl.O=C(NCS)N C1(CN(CCN(C)C)CC2CCCCC2)CC2OC(C)(C)OC2C1 Cc1nc(C)c(C(=O)NCC2CCCC2C(N2CCCCC2CF)=O)s1 N1(C(C2C(C(N)=O)C2)=O)CCN(CC2(O)CC=CC2)CC1 c1(C(C(=O)NC)N(C)Cc2ccc(C(=O)NCCCF)cc2)ccc(Cl)c(F)c1 Cc1occc(=O)c1OCC(=O)N(CC(C)(C)NC(=O)CC(C)C)C C(c1cncc(F)c1)=CC(=O)NC(C1CCCN1C(c1ccc(C(N)=O)o1)=O)C N1(C(C2C(CC)C2)=O)CCC2CN(C(c3ccc(O)cc3C)=O)CCC12 CC1CC2(CO1)CN(C(C13COCC1CN(C(=O)C(N1CCNC1=O)C)C3)=O)C2 C(=O)(C(O)CN1CCCC1)NCC1(NC(=O)CCOC2CC2)CCC1 N1(C(CCSCC)=O)CCC2(CC1)CN(C(C13CC(C1)C3)=O)CC2CO CC(C)CC(C(=O)NC1CCC1CNC(c1cnc(N)cn1)=O)C(C)C N1(C(c2cc(COC)no2)=O)CC2CC(C1)N2C(=O)Cn1nnc(C)n1 C(CC(C)(C)C(=O)N1CCN(C(=O)C(O)C(F)F)C(c2cccc(F)c2)C1)SC Cc1nc(C)c(NC(C2(CNC(=O)CC3CCC(CO)CC3)CC2)=O)[nH]1 c1(OC)cc(C)c(CN2C(C(=O)Nc3cccc(OC)c3F)CC3CC23)c(C)c1 C=C(C)C1CCC(C)=CC1CN.C(C(C)C(C)CC)NC(C1N(C(C=C)=O)CCC1)=O c1(CCC)ccc(C(N2CC3CC3(NC(=O)C(C)(O)CC)C2)=O)cc1 C(=O)(C1=C(Cl)CCCC1)NC(CNC(C=Cc1ccc(CC)cc1)=O)C c1(CC)onc(C)c1C(=O)NCCC(C)NC(=O)C(c1ccc(F)cc1)(C)O Cc1ccc(NC2CC2)c(C(=O)OC(c2ccc(-n3ccnc3)cc2)C)c1 C(=O)(C(CCCC)C(C)C)NCC(C)(C)OCC(=O)N(CCCC(=O)NCC)C C(c1ncccc1C)=CC(=O)NC(CCOC)CNC(=O)CSc1nc[nH]n1 c1(C(N(CC(C)NC(CC2(C=C)CCC2)=O)CC)=O)[nH]nc(OC)c1Cl N1(C(C(CN(C(=O)CC2CCCC(=O)N2)C)(C)C)=O)CCC2(CC2)CC1C c1(C(N2CCC(C(C)NC(=O)CC34COC(C3)C4)C2)=O)nnn2c1CCC2 C(CC)(C(=O)NCC(C1CCOC1)NC(c1cc(C(N)=O)[nH]n1)=O)=CC C(=O)(C1COc2ccccc21)N(C(C)CNC(=O)COC1CC(F)(F)C1)CC C1(C(=O)Nc2cccc(NC(c3cnn(C=C)c3N)=O)c2)CC2CCCN(C1)C2 c1(C2(NCc3nc(C)oc3)CC2)ccc(Br)nc1 c1(N(C(C(C)SCCCC)=O)C)nc(CN)no1 c1(C(N2CCC(N3CCCC(F)C3)CC2)=O)cc(Cl)c(Cl)s1 N1(C(C2C(NC(C3(CC)COC3)=O)CCOC2)=O)CC2(CCOC2=O)C1 c1(-n2c(=O)nccc2)nc(=NCCC=CBr)[nH]c2cc[nH]c12 c1(CC)cc(F)ccc1C(=O)NC1CCC(N(C(=O)CCN2CCCC2)C)C1 C=CCCCC(=O)N1CCSCC1C(=O)NC(c1[nH]c(C)nc1C)C CC1CC(CNC(C2CC2C)=O)CCN1C(=O)CNC(c1ccsc1)=O C(C(CC(C)C)NC(c1csc(C)n1)=O)NC(COCCC#C)=O N12CCN(C(=O)C3CC3)CC1C2=O.Cn1cc(Oc2cn(C)cn2)cn1 C(CCCCCC(=O)NCCN(C)C(=O)C1CC1)N(C(C=C)C(C)CC)C C(=O)(CCC(C(=O)NCC(C(C)(C)C)NC(=O)Cc1csc(C)c1)N(C)C)OC c1(C(C(=O)NCCC(C)NC(=O)Cc2cn(C)cn2)(C)C)ccc(Cl)cc1Cl N1(C(CCCSC(C)(C)C)=O)CCC2(CCN(C(C3C4CNC(=O)C34)=O)C2)C1 C1(NC(C2C(NC(C3(C)CCCC3)=O)COC2)=O)CC2CCCCCC12 N1(C(c2cnc(OCC)s2)=O)CC2CC(C1)N(C(c1ccc(CC)nc1C)=O)C2 CCCC(C(C)(C)C)NC(=O)C(Cn1cccn1)NC(=O)CCC(C)(F)F c1(OC)ccc(OC)c(-c2ccnc(CNC(=O)Cc3cncc(C)c3)c2)c1 N1(C(CNC(CC)=O)=O)CCC(CNC(C23CC(CN2C2CC2)C3)=O)C1(C)C CN1C(=O)CSC1=CC(=O)NC1CN(C(c2ncccc2Cl)=O)CCC12CCC2 C1(CNC(c2cnn(C(F)F)c2)=O)C2CCC(C2)N1C(=O)C(F)F c1(C(N2CCC(N(C(=O)C(C)NS(C)(=O)=O)CC)CC2)=O)cccc(=O)n1C C(=O)(C(O)CCCNC(=O)Cc1cc[nH]n1)NCCC(=O)NO C(=O)(CC(C)C(=O)NC1(C(N2CC3(CC(F)C3)C2)=O)CCN(C)C1)OC c1(C(=O)NC2C(NC(C(CO)OC)=O)CCCC2)ccc(C#N)cn1 C=CCC(C)N=c1nc(N(CCCS(C)(=O)=O)C)c2cc(OC)ccc2[nH]1 S(=O)(=O)(c1cccnc1)NCC(N1CCC(NC(c2cncnc2)=O)C(F)C1)=O Cc1cc(=O)n(CC(=O)N(CCCOCCN(C)C(C2CCOC2)=O)C)cn1 c1(C(=O)NCC(CNC(C2(CC)CC2)=O)C)ccc2c(c1)CCCC2 C(CNC(=O)C=Cc1ccncc1)(CC(=O)NC(C(C)(C)O)C1CC1)OC c1(CNC2C(NC(=O)OC(C)(C)C)C2)ccn(C2CCCC2)n1.OCN c1(C(=O)NCC2(NC(CSCCC#N)=O)CCC2)cccn2cnnc12 N1(C(C(C)SCCCC)=O)CC2CCC(C1)N2C(C12CCCCN1CCC2)=O C=CC1(C(=O)OCCOCCNC(=O)C(=O)NCCCC)CCC1.CCC(N)=O N1(C(CN(C(C)=O)C)=O)CCC(c2cn(CCC(F)(F)Cl)nn2)C1(C)C Cc1cnc(CC(=O)NCC(C2CCC2)NC(=O)C(=O)Nc2ccccc2)s1 c1(C(=O)NCCC2(OC)CN(C(C3(C)CC3(F)Cl)=O)C2)cc(OC)ccc1O c1(OC)cnc(C(=O)N(CC(C)N(C(=O)CC2C=CS(=O)(=O)C2)C)C)c(F)c1 C(=O)(CCC(C)S(C)(=O)=O)NC1(CCNC(CCc2cnc(C)o2)=O)CC1 C(CCF)(C(=O)Nc1ccc(C(C)C)nc1)NC(C(C)NC(=O)C1CC1)=O COn1cnc(C)c1C(N1CCC(C(C)NC(=O)CCc2ccc(C)s2)C1)=O c1(CNC(C(CC)OC)=O)ccc(C(N2CCCC2(C)CO)=O)cn1 CN1CCN(C(C2(C3CC3)CCCO2)=O)CC1C(=O)NCc1csc(Cl)n1 CN1CCN(c2ncc(C(C)(C)O)cn2)C(CNC(C2(C)CC=CCC2)=O)C1 N1(C(c2n[nH]cc2Br)=O)CCN(C(c2ncc(F)cc2F)=O)C(C2CCC2)C1 CN=c1[nH]c(=NCC(C)(C)CO)[nH]c2c1CCCC2.C=CCN(C)CCOC(=N)O C#CCCCCCC(=O)N1CCCC(NC(=O)C(=O)C(C)(C)C)C1 C1(C(=O)Nc2ccc(CC)cc2)(C(=O)NCC(C)C(=O)NC)CCCOC1 C(=O)(C1=CC(C)(C)C1)NC1CCN(C2CCN(C(c3c(CCC)nco3)=O)C2)C1 C(=O)(C1c2ccccc2C2CC1C2)N(CCNC(C1CC1c1cnc[nH]1)=O)CC c1(COC)ccc(-c2nc(C)c(NCC3CCCN(C)C3)s2)cc1 N1(C(C(COC)(F)F)=O)CCN(C(c2cnoc2C)=O)C(CC(F)F)C1 c1(CN(C(CC)C(=O)C2CC2)CC(=O)NOCc2nnnn2C2CC2)ccc(Cl)cc1 N1(CCNC(=O)CC2CCC(=O)N2)CCN(C(c2ncncc2F)=O)CC1 C1(CC(=O)NCCC2(CNC(COCCCCC)=O)CC2)COCCN1CC N(C(=NCCC(=O)N(C)C)NC1CC=CCC1)CC1CCC(CCCC)CC1 c1(OC)cnc(CCNC(=O)C(=O)NCC2(CS(N)(=O)=O)CCC2)nc1 CCC(CNC(=O)CCC1CC1(Cl)Cl)NC(=O)CCOCC1CC1 C=C(C)CC(C(=O)NC(c1ncn(C)n1)C)NC(c1ccc(C#N)cc1)=O C(=O)(CCCCCNC(c1ccoc1)=O)N1CC(CN(C)CC)C1 CC1CN(C(C2CC2c2ccc(Cl)cc2)=O)CC1CNC(c1c[nH]ccc1=N)=O C1(NC(c2c(C)nc(C)o2)=O)CC2CCC(C1)N2C(=O)C(O)C(F)F N1(C(c2ccc(OC)nn2)=O)CCC(C)CC1CNC(=O)Cc1cccc(Cl)c1 C1(NC(CC)C(C)CN(C)C)CC2(CCN(OC(=O)NC(C)(C)C)CC2)C1 c1(C(=O)NC(CN(C(=O)CC(O)C(Cl)(Cl)Cl)C)(C)C)ccn2ccccc12 c1(CNC(C2(C3CCCCO3)CC2)=O)cccc(S(=O)(=O)CC(F)(F)F)c1 C1(CC(=O)NC(C(C)C)(C)CNC(C2CC=CC2)=O)Cc2cc(F)ccc2O1 c1(NC(C2C(C(=O)Nc3c(OC)ncnc3Cl)C2)=O)nc(C)c(Cl)cc1Cl N1(C(C2CC(F)(F)CN2C(c2ccc(Cl)c(O)c2)=O)=O)CCN2C(=O)OCC2C1 c1(OC)cc(C(=O)NCC(F)CNC(C23CC(C)(C2)OC3C)=O)cc(Cl)n1 c1(CC(C)C)ccc(C(=O)NCC2CC(C)N(C(=O)CSCC(N)=O)C2)cn1 CC(C)CC(C(=O)NC1CC12CCC2)ONC(c1cccc(=O)n1C)=O Cc1cc2c(Nc3nc(-c4cccc(-c5cccnc5)c4)cs3)ncnc2s1 CC(C)C(N)(C(=O)NCc1cccc(S(=O)(=O)N2CCOCC2)c1)C(F)(F)F c1(OC)cccc2c1N(C(c1cc(Br)no1)C(=O)NCCSC)CC2 Cc1cccc(C(=O)NC(C(=O)NC2CC2(C)C)C2CCOC2)n1 C(N=c1[nH]cnc(NCc2nc(C(C)C)n[nH]2)c1C)c1cc(C)n(C)n1 N1(C(C2N(C)C(=O)CC2)=O)CC2CC1CN(C(C1CC1c1ccccc1)=O)C2 c1(OC)ccc(C=CC(=O)NCCNC(=O)CCc2ccc(C)cc2)cc1 C#CCCCCC(=O)N1CC2CC1CN2C(=O)C(=O)NC1CC1 N1(C(C2CCC(CCC)CC2)=O)CC2CC(NC(=O)CNC(=O)NC)C(C2)C1 C1(CNC(c2nc(CC)oc2)=O)CCCCN1C(C1CC=CC1)=O C12(NC(c3c(CC)n(C)nc3)=O)CCCC1N(C(c1ccc(F)c(C)c1)=O)CC2 N1(C(CCC)=O)CCN(CCCNC(C2(C)C=CCCC2)=O)CC1 c1(OCC)ccc(C(N2CCC(NC(=O)CC3CCC3)CC2)=O)cc1OC Cc1ccoc1CC1C(c2cn(CC(=O)N(C)C)nn2)C1 N1(C(c2cc(CC)on2)=O)C(CNC(c2cccc(C3(C)CC3)c2)=O)CC2CC12 C1(CNC(C(CO)OC)=O)CC(C)N(C(c2nnn(C(C)(C)C)n2)=O)C1 C12(C(=O)NC3CCN(C(C4CCS(=O)(=O)C4)=O)CC3F)CC3CC(CC1C3)C2 C#CC1(O)CC(C(=O)NC(CC=CC)C(=O)N2CCC(CC(=O)OC)C2)C1 C1(COC)CN(C(=O)CC2(C(F)(F)F)CC2)CCN1C(=O)Cc1n[nH]c(C)n1 c1(-c2cn(CC3OCCN(C(c4ncc(C)o4)=O)C3)nn2)ccnc(Cl)c1N c1(C(C(=O)NC2CC(C(F)F)C2)NC(C)=O)ccc(Cl)c(Cl)c1.C(C)(COC)S N1(C(c2onc(CC)c2C)=O)CC2CC1CC2CNC(=O)CC1CC1 c1(C(N2CCC(CCNC(C(C)OCCC=C)=O)C2)=O)ccc(C#N)o1 c1(CN2CC(C(C)NC(CCC)=O)C2)c[nH]c2cccc(F)c12 N1(C(Cc2cc(C)cc(C)c2)=O)CC2CC1CN(C(=O)C=Cc1cnn(C)c1)C2 CCCC(C)(CC)C(=O)N1CCCC(NC(C)=O)C1.c12cc(n(C)n1)C(=O)NC2 CC1CCC=C1C(=O)N1CCC(CO)(NC(=O)C(C2CCCCCC2)O)CC1 C1(OC)(CNC(=O)C(O)CC(C)C)CCN(C(c2c(Cl)sc(C)c2C)=O)CC1 C(CCCC(F)(F)C(F)(F)F)N.C1(N(C)C)CC(C)(O)CC1=O N1(C(C2CCC(=O)O2)=O)CCOC2(CCN(C(c3ccc(CCO)cc3)=O)C2)C1 N#Cc1cccc(-c2cn(CC(N3CC4CC(F)(F)CC4C3)=O)nn2)c1Br c1(C(CNC(C2CCS(=O)(=O)C2)C)NC(N)=O)cccc2ccccc12 C(CC(C)C(=O)N1CCC(CCOC)(NC(=O)CCCN(C)C)C1)=CCC C1(C)(NC(CC(=C)C)=O)CCCN(C(=O)Cc2ccnc(Cl)c2F)C1 c1(NC2C(CC)CCCC2)ccc(S(=O)(=O)N2CCc3c[nH]nc3C2)cn1 c1(OC)nscc1C(=O)NC(CNC(c1cc(-c2ccccc2)[nH]n1)=O)C1CC1 CN1CCOC(C(=O)NC2(CN(C(=O)CCOC3CCCOC3)C)CC2)C1 CC(C)(O)C#CC(=O)NC(C(=O)NCCC1(C)CCCC1)C1CCCO1 c1(C(=O)NC(CC=C)CNC(c2ccsc2)=O)cc(C)nc(C)c1 C(C)(CC(=O)N1CCCC(O)(CCNC(c2cnsn2)=O)C1)(C(F)F)N(C)C C(CC(C)(C)CNC(c1cc(C2CC2)cs1)=O)NC(C(c1ccc(N)cn1)C)=O C(=O)(CC1CC(=O)Nc2ccccc21)N(C)CCNC(C1CCC1(F)F)=O C(=O)(C(CC=CCl)c1ccccc1)NC(C)CCNC(c1[nH]ccc1C1CC1)=O CC1C2CC(C(=O)N(C3CN4CCC3CC4)C)(C2)N1C(=O)OC(C)(C)C c1(CN2CCC(CC(=O)Nc3nc(Br)cs3)C2)cc(Br)cc(F)c1F C(=O)(N=c1nc(C(F)(F)F)[nH]s1)N(C(Cc1c(C)cccc1)C)C C1(C(=O)NC(C(C)O)(C)C)CC(NC(C2CCCN2C(C)C)=O)C(O)C1 CC(C)C(C(=O)O)NCC(c1ccc(Br)cc1)c1ccccc1 c1(C(=O)NC(CC(=O)NC(CC)COC)CC2CC2)cccc(O)c1F c1(C(N2CCN(C(c3ccc(C)o3)=O)C(C)C2C)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(C(C)OC(c2cccc(C(=O)OC)n2)=O)=O)ccc(C(F)(F)F)c(F)c1 N1(C(c2ccc(C(F)(F)F)c(Cl)c2)=O)CCC2CN(Cc3ccco3)CC2C1 N1(C(c2c(N)cccn2)=O)CCCC(NC(c2coc(C(F)F)n2)=O)CC1 Cc1nsc(C(c2nnnn2C2CCCCC2)NCCn2cc(CO)nn2)n1 CCC(CC)CCC(=O)NC(C)CCN(C)C(c1ncoc1CCC(F)(F)F)=O CC1(C)CC(NC(C2CC3C=CC2C3)=O)CCN(C(=O)COC2CC(F)(F)C2)C1 CC1CN(C(c2c[nH]c(Br)c2)=O)CCC1NC(=O)C(C1CCCCC1)O C1(C(N2C3CC(NC(C4CNC(=O)O4)=O)CC2CC3)=O)CCc2ccccc2C1O CC1(C)CN(C(=O)CC(C2CC2)NC(c2coc3c2COC3)=O)CCS1 N1(C(CC(C(C)C)C)=O)CC(C)N(C(c2nc(C3CC3)ncc2Cl)=O)CC1C N1(C(CCc2ccc(OCC)cc2)=O)CC2CCN(C(=O)C(N)=O)C2C1 c1(C(=O)NCC2CCN(C(CCC=CC)=O)C2)ccc(C2(C)CC2)cc1 CC(CC(=O)NCCOCCN(C)C(c1cc(O)nn1C)=O)CC(C)(C)C c1(C(=O)NC2CCC(NC(C3(CCC=C)CC3)=O)CC2)c(C)cncc1C c1(C(N2CCCC(NC(CCC(C)OCC)=O)C2)=O)cc2c(o1)CCCC2 N1(C(C(CC)C)=O)CC(NC(=O)Cc2cnsc2)CC2(CCOCC2)C1 c1(-c2cn(CC3C(C(=O)NC4C(C)(C)C4)CCC3)nn2)ccccc1F C(CCC(O)C(=O)NCC1CCC2(CC2)CO1)NC(CS(N)(=O)=O)=O c1(OCC(=O)NCC(CN(C(CC(C)OC)=O)C)(C)C)cc(C)ccc1Cl C(=O)(C1=CCCC1C)NCCC(CNC(=O)C1=CCC1)OC C1(c2ccccc2)CC(C(=O)OC)CCN1C(=O)NCC1CC(C(C)C)C1 Cc1cc(Br)c(S(=O)(=O)NC(C(C)C)c2cccs2)c(Br)c1 O=C(CCC(=O)c1ccc(Cl)s1)NC1CC1NC(c1cnsn1)=O CC(C)(C)C(C#N)C(=O)N1CCCC(NC(=O)C(=O)Nc2ccccc2)CC1 Nc1ccc(CCC(=O)N(CCCNC(C2CCCCC2O)=O)C2CC2)cc1F CCC(C)(C#N)C(=O)N1CC(NC(c2cnn(-c3ccccc3)n2)=O)C(O)C1 N1(C(=O)OC(C)(C)C)CC(CNC(C2CC(P(C)(C)=O)CO2)=O)CC12CCC2 C1(OC)CC(CNC(c2ccc(F)cc2)=O)N(C(=O)CCc2ccon2)C1 c1(C(=O)NCCOC2CN(C(C3CC3Cl)=O)C2)cncc(-c2ccccc2F)c1 CC(CCC(=O)NC1CCCC(CNC(=O)CN(C)CCO)C1)N(C)C c1(CC(=O)NCCC(C)NC(c2cnn(C)c2F)=O)ccc(Br)cc1 c1(C(=O)NC2(C)CN(C(C(CC)=CCCC)=O)C2)cc(Cl)ccc1SCC c1(CC)ccnc(C(=O)NC(CCNC(=O)C(F)n2cccn2)C(C)C)c1 C(=O)(C1CCc2ccccc21)N(C1CCCN1C(=O)CNC(=O)NC1CC1)CC C1(NC(COCCCC(C)C)=O)CN(C(c2c[nH]c(=N)o2)=O)CC(F)(F)C1 N1(C(C(COC)OC)=O)CCC(C(C)C(=O)N(C)CCOCCO)CC1 c1(OC)c(C(=O)NC2CC2CNC(c2ccc(C3(O)COC3)cc2)=O)cnn1C C1(=CC(N2CCC(C(C)NC(=O)C(C#N)C3CC3)C2)=O)CCC(C)(C)CC1 C(=O)(CCC1=CCc2ccccc21)NC1CC(NC(C(CC)SC)=O)C1 N1(C(c2ccc(CC(=O)NC)cc2)=O)CCCCCCC1C(N)=O n1(C(C)C)ccnc1C(=O)NCC(C)(C)CC1CN(C(=O)COc2ccon2)C1 Cn1cnn(CC(=O)NC2CCCC2C(N2C(CO)CC2CO)=O)c1=O N1(C(c2cc(=N)[nH]cc2)=O)CCC(NC(C2CCCS(=O)(=O)C2)=O)CC(O)C1 C1(NC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CC1O CC(=Cn1ccnn1)C(=O)NCC1COCC1NC(C1(n2cnnn2)CC1)=O c1(OC)ccc(F)c(C(=O)N(CC(C)NC(=O)COC2(C)CCC2)C)n1 c1(NC(=O)C(N2CC(CO)OC(C(F)(F)F)C2)=O)cccc2c1OCC2 c1(C(=O)NC(C2CCCN2C(=O)C(C)(C)CF)C)cc(Cl)ccc1-n1cccn1 S(=O)(=O)(c1ccc(Cl)c(C(F)(F)F)c1)N1C2C(NC(C(C)C)=O)CC(CC2)C1 c1(CC(=O)OC)cnc(NC(=O)NCCC2(C)CC2(Cl)Cl)nc1 n1(CC)cc(Br)c(C(=O)NCC2CC(NC(=O)C(O)c3ccsc3)C2)n1 N(C1CCSc2ccccc21)C(=O)Nc1cc(C)c2c(n1)cccc2 n1(Cc2ccccc2)cc2ccccc2n1.N12CCC(C13CC3)Nc1cc2ncn1 c1(C(=O)NCCC2CCN(C(c3c(CC)onc3)=O)CC2)ncc(C)cc1F c1(C(N(CC(C(=O)N(CC(O)CF)CC)C)C)=O)cc([N+](=O)[O-])n[nH]1 N1(C(C(=O)NC(CC)(C)C)COc2ccccc2)CC(CC(F)(F)F)OC(C)C1 C1(C(=O)NC2CN(C(CCCOCC)=O)CC2C)COC(C)(C)CO1 c12cc-1ccc2F.N1(CC(=O)ON)CCC(c2ccc(F)cc2)CC1 C(CCN(C)C(c1ccc(=O)oc1)=O)(C(C)C)NC(C1N(C(C)=O)CSC1)=O c1(C(=O)NC2CN(C(C(C)n3cccc3)=O)CC(C)C2)cc2cccnc2[nH]1 N1(C(C=C(CCC)CCC)=O)CC2CC(C1)N(C(=O)C=Cc1cccnc1)C2 N1(C(C=Cc2nnn(C)n2)=O)C2CCC1C(F)C(NC(=O)CC1C=CCC1)C2 Cc1nc(C(=O)NCCCCCC2CCN(C(c3nccs3)=O)CC2)c(C)o1 C(=O)(CC(C(C)C)NC(=O)CCCNC(=O)OC)N(CCCC=C)C c1(C(=O)OCC2C(C)C2)c(F)cc(F)c(S(C)(=O)=O)c1F C1(C2(C=C)CCC2)(C(=O)NC2CC(NC(C(C=C=C)C)=O)C2)CCOCC1 c1(C(N(C2CCC(NC(=O)C=C(Cl)Cl)C2)C)=O)cccc(Cl)c1O C1(CC(N2CC(CNC(c3n(C)ccn3)=O)C(C(F)(F)F)C2)=O)OC(C)(C)OC1=O C(=O)(CC(C)(C)C(F)(F)F)N1CC2C(CNC(CCC(=O)N(CC)CC)=O)(C2)C1 c1(C(N(C(C2CCCOC2)CSC)CC)=O)ccccc1.c1(CC)cn(CC2CC2)nn1 C1(OC)CC(NC(c2csc(C)n2)=O)CN(C(=O)Cc2cc(C)cc(C)c2)C1 c1(C(=O)NC2CCC(CC(N3CC4C(C(=O)OC)(C4)C3)=O)C2)cc2ccccn2c1 Cc1nn(C)c(C)c1CC(C)C(N1CCN(C(=O)Cn2nccn2)C(CF)C1)=O c1(NC(=O)CCNC(=O)OCC2CCCC2)cccnc1SC1CCOCC1 c1(C(=O)NCC2(CC(=O)NCC(C)C#N)CC2)c[nH]c(=S)cn1 c1(C(=O)NCC2CN(C(c3c(OC)c(C)ncn3)=O)C2)sc2ccccc2c1C C12(c3n(CC(=O)OCC)nc4c3CCCC4)CCCCC=C1OCC2 c1(C(N2CCN(C(CCOCC#C)=O)CC2CC#N)=O)ccc(Br)c(C)c1F N1(C(CCCS(C)(=O)=O)=O)CC(CO)C2(C1)CN(C(=O)CCc1nc(=N)[nH][nH]1)C2 N12CCN(CC1)C(=O)N(C(CC)C)C(=O)C2C.c1(C)cc(-c2ccccc2)ns1 c1(C2C(C(N3CCC(N(C(C(N)=O)=O)CCO)C3)=O)C2)ccc(F)cc1F c1(CNCc2ccc(-c3ccc(C#N)o3)cc2)cc2ccccc2nc1O Cc1cc(C(=O)NC2CC(C)N(C(=O)C3=NOCC3)C2)ncc1C(N)=O N1(C(c2cccn2CC)C(=O)NCCOCC)CC(C(N)=O)CC(C)C1 c1(C(=O)NCCN(C(=O)CN2C(=O)CCCC2=O)OCC)ccc(NC)c(O)c1 c1(OC)ccc(F)cc1C(F)(F)C(=O)NCC(CO)NC(=O)CCCSC C1(CNC(C=CC)=O)(CO)CC12CCN(C(c1cncc(OC)n1)=O)CC2 C(=O)(C1CCCc2n[nH]cc21)NC1C2CC(NC(C3CC(C)(F)C3)=O)C(CC2)C1 c1(C(CC)C)nc(-c2ccc(-c3ccc(F)cc3)cc2)n(Cc2ccccn2)n1 Cn1nc(C(=O)NC2CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2C2CC2)ccc1=O N1(C(C2(OC)CCC2)=O)CCCC(N(C)C(c2coc(Cl)n2)=O)CC1 Cc1ccc(C(=O)NCC2(CNC(=O)CCCC(C)C)CC2(F)F)c(N)c1 N1(C(c2n(C)ncc2CO)=O)CC2(CC2)CC1CN1C(CO)CCC1C1CC1 c1(C(N2CC(c3ccc(C)s3)OCC2)=O)cc(F)c(F)cc1N N1(C(c2ccc(OCC)cc2)=O)CC(O)C(O)C1CNC(=O)Cc1c[nH]nc1C C1(C(=O)Nc2cn(CC)nc2C)CC(NC(=O)C(C)CC2CCC2)C12CCC2 c1(C(N(CC(=O)NCC(C2CCCC2)C)C2CC2)=O)cc(C2CC2)on1 C1(C)(C(N2CCC(CCC(=O)NCC(C(C)C)O)C2)=O)CCCOC1 CCC(C)CCC(=O)N1CC(O)CC1CNC(=O)CNC(c1ccsc1)=O CCCCC(C)CCC(=O)NC1(C(N2CC(O)C(O)C2)=O)CCC(C)(C)C1 C12(NC(c3cccc(C)c3)c3n(CCCSCC)nnn3)CCC(C)(C1)OC2 c1(CN2CC(NC(CCC=C)=O)C(F)(F)CC2)cnc2ccc(Br)cn12 c1(NC(CN(CC)CCCN(C)C)=O)ccc(OC)c(C(F)(F)F)c1 CCC(C)C(O)CC(=O)N(C1CCN(C(=O)CSC)C1)CC c1(N2CCCC(NC(c3c(C(F)(F)F)cc(C)o3)=O)C2)nc(C)cc(C)n1 C12(CNC(C(C)C#N)=O)CC(NC(=O)CCC3NC(=O)NC3=O)(C1)C1(CCC1)O2 c1(C(=O)NC2C(C)CN(C(=O)COc3cccnc3)CC2)cnc2ncccn12 N1(C(c2cc(C)cc(F)c2F)=O)CC2CCN(C(=O)C(C)CCC(C)C)CC2C1 C(=O)(CC(C(C)C)c1ccc(F)cc1)N1CC(COC)OCC1 N1(C(C)C)CCN(C(c2cc(SC(c3cnsn3)C)nn2C)=O)C(C)C1 N1(C(Cc2ccc(C)cc2)=O)CCC(C)CC1C(=O)NCCc1cc(C)n(C)n1 N1(C(CCCN(C)C)=O)CC2(CCN(C(c3ccc(O)c(F)c3)=O)CC2)C1 C1(CNC(=O)CCc2nc(O)n[nH]2)CC(C(=O)NCC#CC2CC2)=NO1 CC(C)CC(Cn1cc(CC2CCCOC2)nn1)NC(=O)CCC#N N1(C(CCS(C)(=O)=O)=O)CCCC2(CCCN2C(=O)C(c2ccc(Cl)s2)=O)C1 Cc1ccc2c(C(=O)NCC3(F)CC(CNC(=O)C4CC4)C3)csc2c1 N1(C(C2(C)COC2)=O)CCC2COC(CNC(c3n[nH]cc3N)=O)C2C1 c1(C(=O)NC(CCCC)CCCC)cc(F)cc(C)c1N C(=O)(CC(O)CNC(=O)CC1CCCN(C(C2(C)CCC2C(C)C)=O)C1)OC C=CCC(C)(C)CC(=O)N1CC(O)CCC1C(N1CC(S(N)(=O)=O)C1)=O c1(C(=O)NC2CC(CNC(C(CCSC)OC)=O)OCC2)cc2ccccc2[nH]1 C1(NC(=O)CCc2ccnc(Cl)c2)CC2CCC1N(C(=O)C=Cc1ncc[nH]1)C2 c1(NC(C23C(CN(C(C(C)n4cccc4)=O)C2)C3)=O)nc2ccccc2[nH]1 CC(C)CS(=O)(=O)CC(=O)NC12CC1CN(C(c1cc(F)ccc1O)=O)C2 c1(C(=O)NC2CC(CC(N3CCCC(CC)C3)=O)C2)ccc2[nH]ccc2c1 CC(=O)C(C)CC(C)C(=O)NC(C1(C(=O)N(C)Cc2cc(C)on2)CC1)C Cc1cccc(C(=O)NC2CC2C2CCCC2)c1I c1(OC)cccc(C(=O)N(C)Cc2ccccc2SCCCO)n1 CCC(C)CCCC(=O)NCCN(CCOCCO)C(C1CC1c1ccsc1)=O C=C(Cl)C(C)(C)C(=O)N1CCC(NC(c2cn(C3CC3)nn2)=O)C1 c1(C(=O)NC(CC)CNC(=O)C(C)NS(=O)(=O)CCC)ccc(C(C)=O)c(F)c1 C1(NC(CC=CCNC(CCn2c(C)ncc2)=O)=O)C(C)(C)C1(C)C CC(C(=O)NC12CC(C1)N(C(=O)COCCc1ccccc1)C2)S(C)(=O)=O CC(CCNC(c1csc(CO)n1)=O)CCNC(=O)CS(N)(=O)=O C1(C(=O)NCC(F)CNC(C2(F)CCC2)=O)CCN(c2ccccc2)C1 C1(CNC(c2cc(C)oc2)=O)CN(C(=O)CNC(C2CCC2)=O)C2CC12 c1(C(=O)NCC2CC(C(=O)Nc3c(C)ncn3C)C2)cc(Cl)ccc1F C1(C(=O)NCC=CCNC(C2CCC(CC(=O)OC)O2)=O)CCC2(CCC2)C1 N#Cc1cccc2c(NC(=O)NCC3CCC34CCCO4)n[nH]c12 c1(CC)nccn1C(C)CC(=O)NCC1CCC1NC(=O)Cn1nccc1C C12(CNC(c3coc(Cl)n3)=O)CCC(CC1)N2C(=O)Cc1ccc(Br)cc1 Cc1c(NC(c2c(CNC(=O)CN=[N+]=[N-])nnn2C)=O)cccc1F c1(NC(=O)NCC(=O)N(CC(C)C)CC#C)ccc(C(=O)NC(C)(C)CC)cc1 c1(Sc2c(C(NNC(c3n(C)cc(Br)c3)=O)=O)cccc2)ccc2c(c1)COCC2 CC(C)(C(=O)NCC=CBr)C1=CCN(C(c2ncccc2F)=O)C1 c1(C(=O)NCC(CC(C)C)NC(C(C2CC2)OC)=O)ccc(C)cc1C(C)=O C1(NC(c2ccc(C(=O)OC)o2)=O)CS(=O)(=O)CC1NC(=O)CCCF CCCCC(C)C(=O)NCCCN(C(c1cnn(C)n1)=O)Cc1cccnc1 C(=O)(C(F)(F)CCn1ccnn1)N1CC2C(CNC(C(C)n3cccc3)=O)(C2)C1 C1(O)(CN(C(=O)CCc2cnc(O)[nH]2)C)CCN(C(c2sccc2CO)=O)C1 C1(n2cc(CCN(C)C)nn2)CN(C(=O)CC(C)CC)CCC1C1CC1 N1(C(C(C)(C)CF)=O)CCC(NC(c2cc(O)cc(Cl)c2Cl)=O)C(F)(F)CC1 N1(C(C2CC3CCC3C2)=O)CC2(CCN2C(c2cn3ccnc3s2)=O)C1 Cc1ncc(C(N2CCCC2C(N2CCOCC2)=O)=O)c(Sc2ccccc2)n1 N1(C(CN2CC(C)C2)=O)CCC2(CC1)CC2NC(=O)CCc1cc(F)ccc1F N1(C(=O)C2CC2)CC2(CCC2)CCC1CNC(c1cnc(OC)c(C)c1)=O C1(NC(c2cc(C(C)C)no2)=O)CCOCC1NC(c1ccc(C(F)F)nc1)=O c1(C(=O)NCC(CNC(CSCC)=O)(C)O)ccc(-n2ccc(C)n2)cc1 C12(CNC(C3C(C)OCCO3)=O)CCC(CC1)N2C(C1(CC2CC2)CCC1)=O Cc1ccccc1C1CCN(C(C2CC3(CCC3)C2)C(=O)NC2CC2)CC1 C1(CNC(C(C)OCC)=O)CCC2CN(C(c3ncccc3N)=O)CC12 Cn1ccc2c(CN3CCC(=CC(=O)NCc4cc[nH]n4)CC3)cccc12 N1(C(C2CC=CC(NC(=O)C=CCO)C2)=O)CC2COCC(C2)C1 C(=O)(CCCCCCCO)N1C(C(=O)Nc2cc(C)no2)CCC1 Cc1nc2nccc(C(N3C(CNC(c4csc5cccnc45)=O)CC3)=O)n2n1 Cc1ccc(C)c(C(=O)NC2CC(O)(CNC(=O)CC3CC3C(F)(F)F)C2)c1 C1(CC(=O)NC2CN(C(c3c(C)cnnc3)=O)C2)CCCC(F)(F)C1 C1(N(C(Cc2c(C)n[nH]c2)=O)C)CCC(NC(c2ccsc2C(F)F)=O)CC1 C(=O)(C1=CC2(CCOCC2)C1)NC(C1CCN(C(c2c(SC)cn(C)n2)=O)C1)C CCS(=O)(=O)C=CC(=O)N(C1CC(COc2ccccc2)CO1)CC1CC1 C(CC(O)C(=O)NC1CC1c1nn[nH]n1)NC1(C)CCCC1 N1(C(C2C3N(C(c4nc(C)n(C)c4)=O)C(CC3)C2)=O)CC2(CNC(=O)OC2)C1 C1(CNC(c2c(C(C)C)scn2)=O)CC(C)(C)CN1C(c1ccncc1O)=O FC1(F)C(NC2CCN(C3CCS(=O)CC3)CC2)C12CCOCC2 C1(C(=O)NCCC(C)NC(C2CC(C)(C(=O)OC)C2)=O)COC2(CCC2)C1 C=C(Cl)CC(C(=O)NCC1(F)CCOC1)NC(C1C=CC1C(=O)OC)=O C1(C(N2CCC(C)(F)C2)=O)CCC2(CC2)N1C(C1CC2CCC(C1)O2)=O C1(OC)CC2CCC1CC2C(N1CC2CC(NC(C3CC(C)OC3C)=O)C1C2)=O c1(NCC(CNC(C(CC)C(C)C)=O)O)c(C)c(C)nc2ncnn12 C(=O)(C1=CCC(C)CC1)N1CC(CCCC)N(C(C2CN(C)CC(C)O2)=O)CC1 N1(C(CNS(N(CC(C)C)CC)(=O)=O)=O)CC(C)SCC12COC2 c1(NC(=O)OC(C)(C)C)nc(C2CCCS2)n(Cc2cccc(F)c2)n1 CC(C)CC(O)C(C)C(=O)NCC1(CC(N2CC(N=[N+]=[N-])C2)=O)CC1 c1(C(=O)NCC(CNC(c2coc(CO)c2)=O)CO)ccc2c(c1)CCC2 N1(C(C)=O)C2CCC1CN(C(=O)Cn1cc(-c3c(O)nnc(C)c3C)nn1)CC2 c1(OC)ccc(C(C)NC(=O)C(=O)NC2(C)CCC2)c(NC2CCCC2)c1 C1(CC(=O)NCC2(CSC)CC2)CCCN1C(c1cnn(C(F)F)c1)=O Cc1nn(-c2ccccc2F)c(C)c1NC(C1C(C)C1(F)F)=O c1(CCC(=O)NC(CCNC(C2(F)C(C)OCC2)=O)(C)C)ccc(Cl)cc1Cl N1(C(c2cnc(C)o2)=O)CCC(C=CC(=O)NCCc2cccc(O)c2)CC1 n1(C(C)C(=O)NCC(F)CNC(C2(C#N)CCOCC2)=O)cc2ccccc2n1 C(c1c(F)cccc1F)=CC(=O)NCc1cccc(CNC(c2cncs2)=O)c1 c1(OC)ccc(C(=O)NCC(C)(CC(C)C)NC(c2ccc(C)nc2)=O)cc1Cl CON(CCC(=O)Nc1ccc(F)cc1)C(=O)c1cnc(=N)[nH]c1 N1(C(c2cn(CCOCC)nc2)=O)CCCC1(C)CNC(C1CCCN1C)=O c1(CCC(=O)N(CC(CC)NC(c2cn(C(F)(F)CO)nn2)=O)C)ccncc1 N1CCC(C2CC2)C1C.Cc1ocnc1Cn1cc(CNS(=O)(=O)C2CC2)nn1 C1(NC(=O)CCCN2CCCCC2)CCN(C(C2COCCO2)=O)CC1O Cc1cncc(CC(=O)NC(C)(CNC(c2cnccc2N(C)C)=O)CO)c1 S(=O)(=O)(c1ccc(C)cc1C)Nc1c2ccn(CC)c2ccc1 N1(C(C2(C)CCOCC2)=O)CC(C(=O)NC(CO)CCCO)C2(CC2)C1 C1(C(N2CCC(N(C)C)C2)=O)(CC)CCN(C(C2(c3ccccc3)CCC2)=O)C1 Cc1nc(C)c(C(=O)NC(C)(CNC(C2CCOC2(C)C)=O)C2CC2)s1 c1(C(=O)NCC2C(NC(c3cc(C)c(C)nc3)=O)CCC2)ccc2nn[nH]c2n1 C1(CNC(CCCC(=C)C)=O)CCC2CN(C(C3CS(=O)C3)=O)CC12 C12(CNC(C(C)OCCCC)=O)CN(C(=O)C(=O)N(C)C)CC1CS(=O)(=O)C2 N1(C(c2ccc(C(C)C)cc2)=O)CCC(F)C(NC(c2cc3[nH]ccc3s2)=O)C1 C1(NC(COc2c(OCC)cccc2)=O)CCN(C(C2C3CCCC23)=O)C1(C)C Cc1cccc2c1OC(C(N1CCN(C(C3CCCC3)=O)CC(C)(C)C1)=O)C2 C(=O)(C(C)(C)C(=C)Cl)NC1CC(OCC(N2C(CCC)CCC2)=O)C1 C=CCCCC(=O)N(CCC(=O)NCC1(O)CCN(C)C1)OC C1(C(C2CCN(C(C(C)SC)=O)CC2)NC2(CCN=[N+]=[N-])CC2)CCCC(F)(F)C1 CCCC(CC(=O)NCCC(O)COC)NC(=O)C(C)CO Cc1noc(C)c1C(C)C(=O)NCC1CN(C(c2cscn2)=O)CC1C(F)(F)F C1(CCOC)(NC(C(CCC)N(C)C)=O)CCN(C(C2NC(=O)OC2C)=O)CC1 CCCCC(COC)NC(=O)C(F)CSC.C1(=O)CC(C)N1 C(CC(O)C(=O)NC(C)C(=O)NO)NC(C(c1ccn(C)n1)C)=O C1(C(=O)NCC23OCCC(NC(=O)CC4CCC4)(C2)C3)CCC(=C(F)F)CC1 C(=O)(CC(C)(O)C=C)N1CC(CC=C)(NC(C2CC2C2CCC2)=O)C1 C1(C)(C=O)CCCNC1.CC(C(F)(F)F)N(C)C.c12ccn(n1)CCN(C)C2 N1(C(C2(CC)CCOCC2)=O)CCC(CNC(c2nnc(C)s2)=O)C(F)(F)C1 CC(C)(F)CCC(=O)N1CCC(C)(C)C1C(=O)NCC1(C#N)CCCC1 O=C(C(O)c1ccsc1)NCCNC(=O)CCNC(c1ccoc1)=O C(=O)(CC(=O)NC1CC1)NCC(C1CCOC1)NC(CC1(OC)CCC1)=O C(=O)(C(C)CCOC)N(CC(CNC(C1(CC#C)CCC1)=O)C)C C(CCC(C)NC(=O)Cc1ccnn1C1CCCC1)NC(CSCC=C)=O CN1CCCC1(C)CCN=c1ccn2ncc(S(=O)(=O)NCCCSC(F)F)c2[nH]1 N1(C(C2N(C(c3c(C)ccc(I)c3)=O)CC3(CC3)C2)=O)CCCN2CCCC2C1 CCC1=C(C(=O)NC(CC(=O)N2CCC(O)CC2C2CC2)C(F)F)CCCO1 c1(C(=O)NC(C(C(=O)N2CCNC(=O)C2C)OC)(C)C)cc2ccccn2c1 CC1C(NC(=O)CCc2cn(C)nn2)CCCN1C(=O)CCC1(C)CC1 Cc1c(F)ccc(CNc2cn(C)c(C(=O)NCc3ccc(O)nc3)n2)c1Cl Cc1cc(N2CCOC(C)(C)C2)ncc1S(=O)(=O)NCC1CCC=CCCC1 N1(C(C2C(c3n(C)ncc3)C2)=O)C2CCC1C(NC(=O)COc1cccc(Cl)c1)C2 N1(C(C=C(C)C(C)C)=O)CC2(C(F)(F)F)CC1(C(=O)NC(c1noc(C)n1)C)C2 CCN=C(NCc1conc1C(F)(F)F)NCCC1CCCCO1 C(=O)(C1=NNC(C(F)(F)F)C1)NC1C(C)CN(C(C2CCCO2)=O)C1 CCC(C)(C(=O)NC1CCCCC1NC(=O)C(C)(C)n1ccc(C)n1)C(N)=O C1(NC(C(C(C)O)C)=O)CC2CN(C(c3cnn(CC4CC4)c3)=O)CC12 C#Cc1cnn(C)c1C(=O)NC1CC1NC(c1cccc(Cl)c1Br)=O C1(C(CNC(C2(n3ccnn3)CC2)=O)(C)C)CC(F)(F)C1.C1CCC(=O)N1C c1(NCC(C)SC)ccc(S(=O)(=O)N2CCCC(NC(C)C)C2)cn1 c1(C(=O)NCC2C(C)CN(C(C3CNC(=O)N3)=O)CC2)cccc(N=[N+]=[N-])c1 C1(CCN(CCN(C)CCOC)CC)CCCC(C)C1.c1(N)nccc(C(=O)OC)n1 C(=O)(C(C)(C)C1CCC1)NCCCOCCNC(CCOC(C)=O)=O C=CC1OCCC1C(=O)N(CC(=O)Nc1ccc(C(C)C)cc1)CC N1(C(COC)C)CCN(C(=O)Nc2cc(C3CCCC3)no2)CC1 C(=O)(C=C(Cl)Cl)N1CC(=C(CNC(CN(C2CCC2)C)=O)F)C1 CC1CN(C(=O)Cn2ccc([N+](=O)[O-])n2)CC(C)CN1C(C12CC(F)(C1)C2)=O CCCC(CCC)C(C)(c1nnnn1CC)NC1(C2CCCOC2)CC1 c1(C(=O)NCCCN(C(C)C)CC2(F)CC2C)scc(Cl)c1Cl C1(NC(=O)CC2(CO)CC2)COCCC1NC(c1cncc(CO)c1)=O CC(CC(N)=O)C(=O)NCCCCCNC(C1(C)COCCO1)=O C(=O)(C1=CCCCC1C)N1CCC(N2CCN(c3ncnc(CC)c3F)CC2)C1 N1(C(c2cc(CC)on2)=O)CCN(C)C(CNC(=O)Cc2cnns2)C1 c1(C(=O)NCC(CCCC)NC(=O)CC(C)C(C)C)ccc2c(c1)CCC2(C)C Cc1cc(CNC(=O)C(C)C(C)NC(C2(CO)CCCCC2)=O)ncn1.C(N)(=O)N C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC1CCC(NC(c2n(C)cnc2)=O)CC1 C1(CNC(CC=C)=O)CCN(C(C2CC2C(=O)NCCO)=O)C12CC2 O=C(C#Cc1cccc(Br)c1)NS(=O)(=O)c1ccc(I)s1 C1(CNC(C2N(C(CC)=O)CSC2)=O)C(C)CCN1C(=O)CCc1cnc(C)o1 N1(C(C=C2CCC(C)C2)=O)CCCC2(C1)CN(C(=O)COCC(C)(C)C)CCO2 C12(C(N3CCN(C)C(CO)C3)=O)CCC(CC1)N(C(C1(Cl)CC1(F)F)=O)C2 O=C(C1=CCc2ccccc21)N1CCC(N(C(=O)C(F)C2CC2)CCO)C1 C1(C(=O)NC2(C)CCN(C(CNS(CC)(=O)=O)=O)C2)CC(=O)N(C)C(=O)N1 Cc1cc(=NCCC#CCO)[nH]c(N(CC(C)CN(C)C)C)n1 CC1OC2(C)CC1(C(=O)NCCCCCCNC(C1(CCF)CCC1)=O)C2 C1(C(=O)NCC(C2CCC2)NC(c2c(C)noc2C2CC2)=O)CC12CCSCC2 N1(C(CCCC)=O)CC(COC)CC1NC(c1ccnc(C(C)CC)n1)=O O(NS(=O)(=O)c1cc(Br)ccc1C#N)c1ccc(OC)c(CO)c1 c1(OCC)ncc(CC)cn1.c12nc(co1)CCNC(=O)N2 c1(C(=O)NC23CCCN(C(=O)CC4CC4)CC2C3)ccnc2ccc(O)cc12 n1(CC)ncc(C(=O)N(C)CC2CCCN2C(=O)C(C)(C)C2CCOCC2)n1 c1(C(=O)NC2CCN(C(CCC(C)OC)=O)C2C)cccn2c(C)nnc12 CC1CCC(NC(c2nnc(S)n2C)=O)CN1C(c1ccc(N)cc1Cl)=O N1(C(CCCC=C)=O)CCC2(CC1)CN(C(c1n[nH]c(C)c1C)=O)CC2CO N1(C(=O)Nc2cc(-c3ccccc3)ncn2)Cc2n[nH]cc2C1CO C12(C(=O)NCC3(C)CC(C)(C)C3)CCC(CN(C(c3cnc(C4CC4)o3)=O)C1)C2 C1(C(=O)NCCC2(C(=O)NCCC3C(C)C3)CC2)CN(C)C(=O)N1 c1(C(=O)NC2CC3CC2N(C(C2CCC=CCC2)=O)C3)cc2cnccc2o1 C=CCC(C)(C)C(=O)N1CCC(c2nnnn2C)(NC(C)(CSC)C(N)=O)CC1 c1(OC)ccccc1C(CNC(c1cncs1)=O)NC(=O)C(O)Cn1cncn1 S(=O)(=O)(C1CS(=O)(=O)c2ccccc21)N(CC(F)F)CC C12(C(N(CC)CC3CCCCN3C(=O)CC3CC3)=O)CCC(F)C1CC2 C=C(Cl)CC(C(=O)NC(CCO)C(C)(C)O)NC(c1cc(OC)n[nH]1)=O C=CC(C)(CC)C(=O)NCC(=O)NCC(N1CCC(COC)CC1)=O N1(C(C(CCC)C)C(=O)NC(C)C)CCC2(CC1)CCN(C)C2=O C(=O)(CCCC(C)=O)N(CCN(C(COC)C(=O)NC1CC2CCC1N2)C)C c1(C(N(CC(CC)NC(=O)C(O)CSC)CC)=O)ncnc(O)c1Cl C1(N(C(=O)CC2CCCOC2)CC#C)CCN(C(=O)CCCOCC#C)CC1 c1(C(C(=O)N(C)CC2CC(F)CN2C(=O)CC(F)(F)F)O)cc(Cl)cc(Cl)c1 c1(NCC(N2CC(OCCOC)C2)=O)cnn2ccc(Cl)c(F)c12 C(CN=c1[nH]c(Cl)nc2c1CC(C)CC2)N(C(C(CC)NC(C)=O)=O)CC N1(C(C(C)CN(C)C)=O)CCC2(CC1)CCN(C(C1Cc3cccnc3C1)=O)C2 c1(NC(C(C)(N)C2CCOCC2)=O)ncccc1Sc1cccc(Cl)c1 N(C(=NCCC1SCCS1)NCc1ccnc(C(C)C)n1)C(COC)C CC(C)C(C(C)NC(c1nn(Cc2ccccc2)cc1Cl)=O)NC(C1(C)CC1)=O c1(CC(=O)NC(CC=CC(=O)N(CC(CC)O)C)(C)C)cn(C)nc1C CC(C)(C)C(C(=O)NC1CC1NC(=O)C(C)(C)C1CCCCC1)N1CCCC1=O N1(C(c2c(C)n(C)nc2)=O)CC(CO)C2(CCN(C(=O)CO)CC2)C1 N1(C(C(C)(C)OC)=O)CCCC(N(C(=O)CCN2CCCCC2)C)C1 CC1(C)Cc2cc(S(=O)(=O)N3CCOC(Cc4ccc(F)cc4)C3)ccc2O1 C1(NC(c2ccon2)=O)CN(C(=O)COCC2CCOC2)C2(CCC2)C1 c1(C(=O)NC(C2CCCCC2)C(C)NC(=O)C=C(Cl)Cl)cnc2scnc2c1 c1(OC(CC(CC)OC)=O)ccc2nc(CSC(C)(C)C)[nH]c2c1 c1(C2C(CNC(C(=O)NCCSC3CC3)=O)C2)cc(-c2ccccc2)cs1 c1(N(C)C2CC2)nc(N2CC3CC=CCC3C2)nc2c1CCC2 c1(C(C)(F)F)cccc(C(=O)NC2CCC(NS(=O)(=O)C3CC3)C2)c1 C1(NC(C(CSC)C)=O)CN(C(c2cc(-c3ccn(C)n3)on2)=O)CC1C C(CCCC(C)NC(c1cncn1C)=O)NC(C1(C=C)CCC1)=O c1(N(CCNC(c2c(CC)onc2)=O)C(=O)OC)c(F)cccc1[N+](=O)[O-] CC1CN(C(=O)CCS(C)(=O)=O)CCCN1C(c1c(N)cc(Cl)nc1Cl)=O N1(C(c2c(CC)cccc2)=O)CC2CCN(C(c3cnnn3C3CC3)=O)C2C1 c1(CC(=O)N(C(C)(C(=O)NC)N(C(C(OCC)OCC)=O)C)C)cccc(C)c1 N1(C(c2cc(C)ns2)=O)CC(C)N(C(C2CCSC2)=O)CC1C C1(NC(Cc2cc(OC)no2)=O)CCCCN(C(c2csc(Br)c2)=O)C1 CCC(CC)(CC)C(=O)N1CCCC2(NC(=O)Cc3ccc(O)nc3)CC2C1 Cc1[nH]c2ccccc2c1C(N1CCC(NC(c2cc[nH]c2C)=O)C(C)C1)=O c1(C(=O)NCC2(O)CC2C(F)(F)F)n[nH]cc1CNC(c1cnco1)=O Cc1nc2ccccc2nc1C(=O)NC1CCC2CC1CN2C(C1CC1CF)=O Cc1nc(CCOC(C)(C)C)[nH]c1NC(=O)OCCCNS(C)(=O)=O C1(C(=O)Nc2cc(C(=O)OC)c(Br)cc2)CCCC12CN(C(=O)CSC(C)=O)C2 c1(N2CCC(OC)C(C)(O)C2)ccc(S(=O)(=O)NCCc2cc(Br)cs2)cc1Cl C1(CCNC(C2(C=C)CCOCC2)=O)CN(C(=O)C(C)COC)CCS1(=O)=O Cc1ncnc(C)c1CC(=O)NC(C)C(CO)NC(c1ncccc1F)=O CCCN=C(NCCNC(C1(C)CCCO1)=O)NC1CC(C(=O)OC)C1 N1(C(=O)OC(C)(C)C)CCCC2C1CCCN2C(c1cncc(F)c1C(=O)O)=O Cc1noc(C)c1C(=O)NCC1(NC(=O)C=Cc2cn(C)nn2)CCCCC1 CC1OC2(C(N3CCCC(CN(C)C(C4CC4C(N)=O)=O)C3)=O)CC1C2 C(=O)(C1CCCc2ccnn21)NCC1CC(NC(c2cnc(C)[nH]2)=O)C1(C)C C(=O)(CCCS(N)(=O)=O)NCc1[nH]c(=NCc2nccc(C(=O)OC)c2)sc1 C1(CNC(C(CSC)C)=O)CC(F)CN1C(=O)C=CCN(C)C C1(CNC(CNC(CNC(C)=O)=O)=O)CCN(C(c2csnn2)=O)C1(C)C CC(CC(N)=O)C(=O)N1CC2CC2(CNC(c2cnc(O)c(F)c2)=O)C1 c1(C(C(=O)NCCOC)N(CC(C)C)CC#N)cc(C(C)C)[nH]n1 C=CCC(F)(F)CN=c1nc(N2CCc3ccccc3C2C=C)c2[nH]ccc2[nH]1 CCC(CCC(=O)N1CCC(NC(C2(COC)CCCO2)=O)C1CC)OC CCCCCC(O)CC(=O)N1CC(C)CN(c2ncc(O)c(OC)n2)C(C)C1 CC1(C)CC(CNC(c2cc(Cl)ccc2O)=O)N(C(=O)CC2CCC3CC23)C1 c1(C(N(C2CCN(C(=O)Cc3nncn3C)C2)CCSCC)=O)nn[nH]c1Cl c1(C(N2CC(C)C(NC(c3nc(Cl)ccc3Cl)=O)C2)=O)cc(Cl)c(F)cc1F Cc1cc(CO)oc1C(=O)NS(=O)(=O)CCOC1CCOCC1 N1(C(C(N2C3CC(NC(CCCC=C)=O)(C3)C2)=O)C)C(=O)c2ccccc2C1=O c1(C(N2CC=C(CNC(c3cn(C)nc3)=O)CC2)=O)ccc2cnoc2c1 N1(C(C2CC2c2ccco2)=O)CCCc2nc(CO)ccc2C1 c1(C(=O)NCC(C(C)C)NC(C(C)(CO)NC(C)=O)=O)ccc2ncsc2c1 C1(NC(c2nc(CC(C)C)sc2)=O)CCCC(NC(c2nocc2C(C)C)=O)C1 C1(NC(C2(CCC)CCC2)=O)CN(C(=O)CCS(=O)(=O)NC)CCC1(C)C C(CC1=CCN(C(c2ccnnc2C)=O)CC1)NC(c1cc(OC)ncc1Cl)=O CC(=O)CC(C)(C)C(=O)N1CCC(C)N(C(=O)C#CC(C)C)CC1 N1(C(Cc2c(C#C)cccc2)=O)CC(NC(=O)C(C2CCOCC2)F)CC(F)(F)C1 Cc1ncc(CNC(C2(C)CC(NC(=O)C(c3cncnc3)C)C2)=O)o1 c1(CC)onc(C)c1C(=O)NCc1ccc(C(=O)NCc2cc(OC)n[nH]2)cn1 c1(CC)cc(-c2cccn2CC(=O)O)cc(-c2cnc[nH]2)c1 Cn1cc(NC(C2CCC(NC(c3cnc(NC(C)=O)[nH]3)=O)CC2)=O)c(C(N)=O)n1 c1(C(=O)OC)cnccc1-c1cccc(NCc2n[nH]cc2Cl)n1 CCC(CNC(=O)CCC(=O)NCC(F)(F)F)(CC)OC.C(=O)(CCOC(C)C)N N(C(=NCC(C)C)NC)Cc1cc(OC)ncc1.c1(CSCCO)cccc(F)c1 C1(NC(CCC(C)OCC)=O)CCN(C(c2ccc(CC)c(F)c2)=O)C12CC2 C(=O)(CC1OCCc2ccsc21)NC(CC)CNC(c1cnc(Cl)s1)=O C(=O)(CCCC(F)F)NC1CN(C(COCP(C)(C)=O)=O)C1 C#CCC(C)(CNC(=O)CCCCC)CO.c12ncccc1OC2=O N1(C(CCC=CCCC=C)=O)CCCC1C1CCCN1C(=O)C1=CCSC1 C1(CC(=O)NCC(C)N(C(C2CCCN2C2CCCC2)=O)CC)CCC=CCC1 CC1(C)OCCC1C(=O)NC1CCCC(C(N2CCCCC2CCO)=O)C1 C1(C(=O)NC2C=CC(CNC(C(C)=CC)=O)C2)CCc2nc(C(F)(F)F)cn2C1 Cc1ccc(C#N)cc1NC(=O)C(C1CC1)NC(=O)Cc1cnnn1C Cc1cc(C(=O)N(C)CCN(C)C(C2CCOC2C(F)(F)F)=O)ncc1N C1(NCCNC(c2cn(CCC)nc2)=O)CNCC(C)C1 c1(N(C(C(n2cc(C3(N(C)C)CCC3)nn2)C)=O)CCC#N)ccc(F)cc1 C(CCCC(=O)NC1CCC(CCNC(=O)COC2CC=CC2)C1)(OC)OC C1(C)(C(=O)NCC2(CCOC)CC2)CCCN(C(=O)Cc2cc(C)no2)C1 Cc1ccccc1C(=O)NCC1CCN1C(=O)C=C1CCC1 N1(C(Cc2c(C)noc2Cl)=O)CCCN(C(=O)Cc2ccsc2C)C(CO)C1 C(C)(C(=O)N=c1ccn(CC(C)C)[nH]1)C1CCCN(c2c(C(C)=O)cc(C)s2)C1 N1(C(C(=O)NC2CC2)=O)CC2CCCN(C(c3cnc4c(c3)OCCN4)=O)C2C1 C1(S(N)(=O)=O)(C(N2CCC(CN(C(=O)COCCCOC)C)C2)=O)CCC1 c1(C(N2CCC(N(C(C=CC)=O)CCO)C2)=O)nc(Br)n2c1COCC2 N1(C(C(CC=CC)CC)=O)CC(CO)C2(C1)CN(C(=O)CCN1CCC1)C2 C(=O)(C(C(C)C)c1cnn(C)c1)NC1CN(C(CCC=CC(C)C)=O)C1 c1(C(=O)NC2CCCCC2NC(C2CCO2)=O)c[nH]c2ccc(F)cc12 C(=O)(C(O)C(C)CC)NCCCCNC(C1(CC#C)CC(F)(F)C1)=O C#CC1(C)CCCN(C(=O)C(C)(CSC)NC(c2ccc(O)cc2)=O)C1 c1(C(=O)NCC(C)CN(C)C(c2cc3cc[nH]c3cn2)=O)ccc2c(c1)OCC2 c1(C(=O)NC(c2cccc([N+](=O)[O-])c2)C(=O)O)csc2c(Br)cccc12 c1(C(N(C2CSC2)CC#C)=O)ccc(CNC(C2COC(C)C2)=O)s1 Cc1cc(CNC2CCCN(C(C3(c4cccc(Br)c4)CCC3)=O)C2)ccn1 C1(C(N(CCOCCC(=O)NCC(OC)OC)C)=O)CCC(=O)N1C c1(C(=O)NCC(C2CCN(C(CN(C3CCSC3)C)=O)CC2)O)ccnnc1O c1(C(N2CCC(CC(F)F)CC2)C(=O)NC(C)(C)C)ccc(Cl)c(Cl)c1 C1(C(N(C2CCN(C(c3cc(C#N)on3)=O)C2)C)=O)CCCCC12CCC2 c1(C(N2CC(NC(c3csc(O)n3)=O)C2)=O)ccc(F)c(F)c1 c1(C(N)=O)cc(CNCC2(O)CCN(C(C(CCSC)O)=O)C2)cc(F)c1 N1(C(C(C)C)=O)CCN(C(=O)CCNS(=O)(=O)c2cccs2)C2CC12 N1(C(CC(CC)C)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)C(C)C C1(C(=O)NCCC2CC(NC(=O)CN(C)C(N)=O)C2)(OCC)CCCCCC1 N1(C(C)=O)CCOCC1C(=O)NCCCN(C)C(c1sccc1C)=O c1(OC)nc(NC2CC(NC(=O)Cn3nc(Cl)ccc3=O)C2)ncc1Br C(=O)(CCP(C)(C)=O)N(C)Cc1ccccc1CNC(c1c(Cl)nsc1Cl)=O N1(C(C(C)NC(=O)NC)=O)CC(NC(=O)CCS(C)(=O)=O)CC12CCC2 C(=O)(CC1=CCN(C)CC1)N(CCCNC(c1c(CC)cccc1F)=O)C C(C(CC)n1cccn1)NC(=O)NCCCN(CCC#C)C N1(CC2(C(=O)O)CC(C)(C)C2)CCCCC12CC(CNC(=O)OC(C)(C)C)C2 C(=O)(CC1COc2ccccc21)N1CCCN(C(Cc2c(C)cccc2)=O)CC1 C(=O)(C1=CCOCC1)N(CC(C)O)CCNC(C(CC)OC)=O n1(CC)cc(Cl)cc1C(=O)Nc1ccc(NCCc2ccccc2)cn1 c1(OC)cc(C(N2CC3(CC(NC(=O)C=CC4CCCO4)C3)C2)=O)c(F)cn1 c1(CNC(=NCc2cncc(O)n2)NC2CCC2)cc(I)ccc1Br.CCCC N1(CC)C(=O)CCC1CC(=O)NCC(C)(C)NC(=O)C(C)OCC1CC1 c1(C(N2CC(C(=O)O)C(C(F)F)C2)=O)cccc(O)c1OC(F)(F)F C=CCCC(C(=O)NC1CC(C)(C)OC1=O)NC(c1sccc1F)=O C(=O)(C(CO)C(C)(C)C)NCC1(COC)CN(C(C2C(C)C2C)=O)C1 C1(C(=O)NCC=CC2(C(=O)NC3CCCCCC3)CCCO2)CCC2(CCC2)O1 S(=O)(=O)(c1ccc(N2CCCC(c3ncccn3)C2)c(Cl)c1)NCC(CC)OC c1(CC(=O)NC2CCCCN(C(C(CSC)O)=O)C2)ccc2c(c1)COCC2 N1(C(c2c(OC)ccs2)=O)CC2CCN(C(c3cnn(C4CC4(F)F)c3)=O)CC12 N1(C(C2=CC(C)(C)C2)=O)Cc2n[nH]cc2C1C(=O)NC1CC(C2CC2)C1 C(=O)(CC(C)C(=O)N1C(CC(=O)N(C)Cc2ccn(C)n2)C2CCCC12)OC c1(SCC(N2CCCC(C#C)CC2)=O)c(C)sc2nc(C(C)C)nc(O)c12 Cn1c(=N)[nH]c2cc(C(=O)NC3CC4(C3)CC(NC(C3CCO3)=O)C4)ccc12 C1(NC(C=CS(C)=O)=O)CS(=O)(=O)C2CN(C(c3ccnc(O)c3)=O)CC12 c1(C(N2CC(C(C)NC(c3c(C)cnn3C)=O)OCC2)=O)ccc2snnc2c1 C1(CCC#C)CCCCN(C(=O)CC2CCCCN2C(=O)CN(C)CCC)C1 C(=O)(C1COc2ccc(Cl)cc21)NC(CC=C)CNC(C1CCCCCCC1)=O c1(C(N2CC(NC(c3c(OC)ccnc3)=O)C2)=O)ccc(C#N)c(F)c1Br N(C(=NCCC(=O)N1CCN(CC)CC1)NC1CC2CCC1C2)C(CC)CC CC1CN(C(c2cc(C(F)(F)F)on2)=O)CCC1NC(=O)CSCc1ncc[nH]1 c1(CCC(=O)N(CCOC)CCNC(C2CCC2C)=O)ccccc1F C#CC(C)(C)C(=O)N1CCCC(CC(=O)NC(c2ccc(C)nc2)C)C1 c1(C(=O)NCC(CC2CN(C(C(CC)(F)F)=O)C2)(C)C)cccc2cnnn12 C1(NC(c2cccc(C#C)c2)=O)CCC12CCN(C(=O)CC1C=CCC1)CC2 C(=O)(C(C)N=c1cc[nH]cc1)N(CCCNC(C1CC(O)(CC#C)C1)=O)CC C(=O)(CCCCC(=O)N(C1CC(O)CN(C(=O)CNS(N)(=O)=O)C1)CCOC)NC c1(C(=O)OCC)cc(OC)ccc1-c1csc(N(CC)Cc2ncsn2)n1 C1(NC(CC2C(C)(C)CCO2)=O)CN(C(C2CC3CCC3C2)=O)CC1(C)C c1(C(N2CCN(C3CN(CC)C3)CC2)=O)coc2c1CCCC2.C1(N)CCCC1N c1(CNC(COCCCC)=O)cn(C2CCN(C(=O)C(C)CF)C2)nn1 N1(C(Cn2c(C)nnn2)=O)CCN(CC(C)NC(=O)CC2(C)CCCO2)CC1 C1(C(N2CCC2C2CCC2)=O)(CNC(c2n(C(C)C)cnc2)=O)CC12CCC2 C12(C(=O)OC)COC(C1)C(Nc1ncccc1C(F)(F)F)C2 N1(C(C2(CC)CCCN2C(c2cccc(C)c2O)=O)=O)CC2(CNC(=O)C2)C1 Cc1cc(F)cnc1C(=O)NCc1nc(C(=O)NC2C(O)CC2O)co1 c1(C(N(C)CC2N(C(C3C(OC)(OC)CC3)=O)CCCC2)=O)cncc(C)c1Cl C1(CNC(c2c(C(=O)OCC)con2)=O)CN(C(=O)C(C)CC)CC2(CCC2)C1 N1(C(C(C)OC2CCCC2)=O)CCC(CO)(NC(c2cnc(S)n2C)=O)C1 C(=O)(C(C)CC(C)(C)C)N1C(C(C)C)(C(=O)NCc2c(C)n[nH]c2)CCC1 C1(C(N(C(CNC(c2c(CC)scc2)=O)C2CC2)C)=O)Cc2ccccc2O1 C1(C(N2CCCC(NC(c3cnnc(O)c3)=O)C2)=O)CC(C2CC2)=NO1 c1(C(=O)NC2C(C(=O)NCC3(CC)CCCO3)CCCC2)ccc(C)cc1F N1(c2ncc(C)cn2)CC(NC(C2CCCC23CC3)=O)CCC1C C(=O)(CC1=NNC(=O)C1)N1CCC(C(C)(C)CNC(=O)CC2CCCCO2)CC1 CC1CC(NC(c2cc(=N)[nH]n2C)=O)CN1C(=O)CCCCC1CCCCC1 C1(NC(CC2ON=C(C)C2)=O)CCN(C(c2c[nH]c(=N)c(C)c2)=O)CC1O N1(C(c2ccn(CCC)n2)=O)CC(NC(=O)C(C)CCO)C(C)(C)C1 N1(C(C2COC(C)C2)C(=O)NC)CCC(OCCCO)CC1 C1(NC(CCSCC)=O)CC(CNC(C2CN(CC)C(=O)N2)=O)C1(C)C C(=O)(CCCCCCBr)N1CCCC(C)C1C(F)(F)F C1(C(=O)NCCC(=C)CNC(=O)C(F)(F)c2nccn2C)CCCC(O)C1 Cc1cccc2c(C(=O)NC3CCN(C(c4sc(F)cc4Cl)=O)CC3C)coc12 c1(OC)cc(C(N2CCC(C(C)NC(c3cc(C)nn3C)=O)CC2)=O)cc(F)n1 C(=O)(C1=CCSC1)N1C(CC(=O)NC(COC)CO)CC1 c1(CC(=O)NCC2CC(NC(COC)=O)C23CCC3)c(F)cc(OC)cc1Cl C(C(C)(O)C(=O)NCC1COCC1NC(=O)CCCN1CCCCC1)OC C1(CC=C)CCCCN1c1cc(N2CCC(C(C)C)(CO)C2)ncn1 CC1CCCC(O)(C(=O)NCC2(O)CN(C(c3cnc4[nH]ncc4c3)=O)C2)CC1 Cc1cc(Br)ccc1C(C)C(=O)NC1CCN(C(=O)C(C)(C)C)CC1 C1(CC(=O)NCC2(C(=O)NC(c3ccoc3)C)CCCC2)C(C)(C)C1(C)C C1(C(N(C)CC2CCN(C(Cc3cnc(C)s3)=O)C2)=O)CCC(=O)N(C)C1 Cc1ncc(C(=O)NC2CCC2CNC(=O)CCC2(C)N=N2)c(C(C)C)n1 Cc1ncc(C(=O)NCCC(C)N(C(=O)CC2COCCO2)C)cc1N C=C1C(C(=O)N(CC(CC)NC(C2(C(=O)OC)COC2)=O)C)C1C(=O)OC c1(CC(=O)NCC(C)CNC(c2cc(C(C)(C)C)n[nH]2)=O)cnc(N(C)C)nc1 Cc1cc(C(=O)NCC2(NC(=O)CCn3cc(Cl)cn3)CC2)cnc1F C1(C(=O)NC(CC(=O)OCC)C)C(C)OCCN1C(=O)C(C)CC1CC1 Cc1cc(I)ccc1NC(=O)NC1(Cc2cnsc2)CC1 c1(NC(=O)CSc2nc(C3CCCCC3)no2)ccc(Cl)cc1Cl Cc1c(-n2nccc2NC(=O)NC(C)COc2ccccc2)cccc1Cl N1(C(C(=O)NC(C)C)=O)CCC(F)(CNC(C2CCN2C2CCCC2)=O)C1 CCC(F)(C(=O)OC)C(=O)N(CC(O)CN(C(=O)C(C)(C)C1CCC1)C)C C1(NC(CC(C)(C)C)=O)CC2CN(c3nc(C(F)(F)F)ns3)CC2C1.C1C(=O)N1 C(=O)(CCCN=[N+]=[N-])NCC(CCNC(C1(CCCC)CC1)=O)O C12(C(=O)NC3CCCCC3NC(C3CC34CCC4)=O)CC3CC(C1)CC(O)(C3)C2 C1(NC(C(CC)OC)=O)(CC)CCCN(C(c2cncc(Cl)c2C)=O)C1 c1(CC(=O)NC2(C)CCN(C(C=CCOC)=O)C2)ccc(F)cc1F c1(C(=O)NC(C2CCN(c3nc(C)nc(O)c3)C2)C)ccc2c(c1)OCC2 c1(C(N2CCC(C)(NC(C3CCC(C)(C)O3)=O)CC2)=O)cncc2ccccc12 N1(C(C(C)N2CCC2)=O)CC(C)(C)CC1CNC(c1coc(N(C)C)n1)=O CC1(C)CC(=O)C=C(c2cccc(C(=O)NCCCC(=O)NC3CCCC3)n2)C1 CC(C)(C)C(O)C(=O)N1CCC(OCCNC(c2ccn(CC(F)F)n2)=O)C1 N1(C(=O)NCCc2cc(O)cc(F)c2)CCOc2cc(F)ccc2C1 N1(C(C2(F)CN(C(CN(C3CC3)CC)=O)C2)=O)CCCC(F)CC1 C1(NC(C2C(CN(C)C)C2)=O)CCC2(CC1)CN(C(c1ccc(F)o1)=O)CCO2 C(=O)(NN1CCCC1C(=O)NC1CC2(CCOC2)C1)C1CC2(CC(OC)C2)C1 c1(NC(C(CNC(Cc2c(C)ccs2)=O)O)=O)ccc2occc2c1 C1(CC(=O)NCCC(C)NC(c2cnccc2N(C)C)=O)CC(C)(C)OC1=O C1(NC(c2ccc(NC(=O)OCC)o2)=O)CCN(C(c2cccnc2)=O)CC1C C1(C(=O)OC)CC(F)(F)CN1C(C1CN(C(c2ccc(Br)nc2C)=O)CCN1)=O Cc1cnc(CCC(=O)NC2(CF)CN(C(=O)CCc3csnn3)C2)[nH]1 n1(CCC=C)cc(CC(C)(C)SC)nn1.C1(=O)C(=O)N2CC(C2)CN1 c1(C(=O)NCC(S(C)(=O)=O)CNC(c2cccc(F)c2)=O)csc2c1CCCC2 N1(C(c2c(C)nnn2C)=O)CCC2(CCOCC2)C(CNC(=O)CN(C)C)C1 c1(OCC(=O)N(C(C)CSc2cnn(C)n2)C)ccc(C2CCCS2)cc1 C(c1ccc(Cl)nc1)=CC(=O)NC1(CNC(C2(C(F)(F)F)CCCC2)=O)COC1 C1(N(C(C(Cc2c(C)nc[nH]2)O)=O)C)CN(C(c2c(C)ncn2O)=O)CC12CC2 CCCCCC(F)C(=O)N(C)CC1CCC(NC(C2(CO)CCCO2)=O)CC1 N1(C(c2ccc(OCC)cc2)=O)CC2CC(C1)N(C(=O)CN(C)S(N)(=O)=O)C2 Cc1nc2cc(C(N3CCCC(CNC(C4CCC(C)(C)C4)=O)C3)=O)ccc2o1 N1(C(CCc2ccnc(C)n2)=O)CCC(C)C(NC(c2sc(O)nc2C)=O)C1 Cc1cc(N)c(C(N2C3CCC2C(CNC(c2ccccc2C)=O)C3)=O)cc1F C(=O)(CCC(=O)N1CCC(CCN)CC1)NCC.N1(CCC(=O)N)CCCS1(=O)=O N1(C(c2cn(CC)nn2)=O)CCC(N(C(=O)C(C)n2cccn2)CCO)CC1 C1(NC(C(C2(O)CCCCC2)CC)=O)CN(C(=O)Cn2cnnc2O)C(C)(C)C1 CC(CCc1ccc(F)cc1)C(=O)NC1CC(CNC(C2CCC(O)C2)=O)C1 c1(OCC)cc(C)nc(N2CCNCC2C(=O)NCc2cc(F)cc(Cl)c2)n1 N1(C(C(COC)OC)=O)CCCC(O)(CN(C)C(c2cnn3c2OCC3)=O)C1 C1(CNC(c2ccc(OC)s2)=O)CCN(Cc2cc(Cl)c(O)cc2O)CC1(F)F Cc1cc([N+](=O)[O-])ccc1C(N1CCCC1C(N1CCCC1CO)=O)=O C1(CC(=O)N(CC(CC)OC)C)C2CCC(C2)N1C(c1cccc(CO)c1)=O C1(NC(c2c(C)cc(CO)o2)=O)CCN(C(c2c(Cl)cnn2C(C)C)=O)CC1C c1(C(N(C2CCN(C(C(C3CCC3)OCC)=O)C2)C)=O)csc2c(F)cccc12 C1(NC(Cc2nc(C(C)C)sc2)=O)(CO)CCCN(C(=O)C(O)C(F)F)C1 C1(F)(CNC(C2=NNC(=O)CC2)=O)CC(N=c2[nH]nc(C3CC3)s2)C1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2CC2(NC(=O)C2=CCCS2)CC1 Cc1ccc(CC2CC2)cc1I.c1(C(N(C=O)C)C2CC2)ccccc1 CC1CCC(n2nc(CC3CCOCC3)nc2-c2csnn2)CC1 c1(OCOC)ccc(O)c(-c2cnc(NC(C3CC(O)C3)=O)s2)c1 C(=O)(CC(C)(C)O)N1C(CN(C)C(C2CC2c2cccs2)=O)CCC1 c1(C(N2C(C)CN(C(Cc3c(C)con3)=O)C(C)C2)=O)[nH]c2ccc(Cl)cc2c1Cl c1(C(N)=O)cc(=NC2CCCN(C(c3cnc[nH]3)=O)C2)[nH]c(Cl)n1 C1(C(=O)NC2(C)C(C)(C)C2)CCN(C(=O)CC(C2CC2)C2CC2)C(C)(C)C1 O=C(N=c1[nH]nc(CC2CC2)s1)NCC(c1ccccn1)C1CC1 CC1CC(NC(=O)CNC(=O)CN(C)C)CN(C(c2cn3c(n2)CCC3)=O)C1 c1(C(=O)NCCC2(O)CCN(C(C34CC(C)(C3)C4)=O)C2)c(F)ccc2occc12 C1(C(C)NC(C2CC2C)=O)CCCCN1C(c1nncn1C)=O CCCCCC(C)NC(c1cccnc1CNC(c1ccncc1F)=O)=O N1(C(CC(CC2CC2)NC(C(CC#C)O)=O)=O)CCCC2CCCCC12 c1(C(N2C3CN(C(CCCNC(=O)OC)=O)C(C3)C2)=O)nn(C)cc1S(N)(=O)=O Cc1cc(N2CC3CC2CN3C(c2c(F)cccc2Cl)=O)nc(C(F)(F)F)n1 C=CCC(CNC(c1cnnc(C)c1)=O)C(=O)NC(C(F)(F)F)C1CC1 N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(c2cn[nH]c2)=O)CC12CCCC2 C1(CNC(Cc2c(C)noc2C)=O)CN(C(=O)CC2CC(C)C2)CCC1C C(=O)(C(O)CCCNC(c1ccc(O)c(F)c1)=O)NCC(C1CC1)SC c1(C(=O)NC(CNC(CCOCCC)=O)C(C)C(C)C)cccc2c1CNC2=O c1(C(N2CC(CCNC(C(C)SC)=O)OCCC2)=O)cc([N+](=O)[O-])c(N)cc1F C(=O)(CCCCCNC(=O)CN1CC2CC2C1)NCc1[nH]nc(CC)n1 c1(C(=O)NCC(C(=O)NC(COCC)C)N(C)C)ccn(C)c(=O)c1 c1(SC)ccc(-c2nc(C)nn2C(C)Cc2ccccc2)cc1C N1(C(C(CC)(C)CNC(C2CC(F)C(=O)N2)=O)=O)CC2COC(=O)C2C1 c1(C(N(C2CN(C(CC=C(C)C)=O)CC2F)C)=O)cn2cnnc2cn1 C(CCC(C)CC(=O)OCCCN1CCCC1)=C(C)C C[S+](C)CCC(O)C(=O)NCC(C1CCCC1)NC(c1ccc(C(C)=O)nn1)=O C1(NC(C(CC)SC2CCCC2)=O)CCC(C(=O)NCCN2CCN(C)CC2)CC1 N1(C(Cc2cnc(C)s2)=O)CCOCC1CC(N1CC(F)C(F)C1)=O C1(CC(=O)N(C(C)CO)CC2CCOC2)CCC=CCC1 c1(C(=O)NCC2CCCC(CNc3cc(OCC)ncn3)C2)cc(Cl)ccc1F c1(C(=O)NC2CCN(C(CC(C)C)=O)C2)cc([N+](=O)[O-])ccc1Br C#Cc1cc(C(=O)N(C(C)CNC(c2cncc3c2CCC3)=O)CC)cc(N)c1 c1(N2C(CNC(c3cc(Br)cc(Br)c3F)=O)CCC2)ncnc2c(F)cccc12 c1(C(=O)NC2C3CC2N(C(=O)C(O)C(F)(F)F)C3)ccc([N+](=O)[O-])c(O)c1 c1(OC)ccc(C(=O)NC(CNC(c2cc(C)n(C(F)F)n2)=O)CO)c(F)c1Cl C(=O)(C#CC1CCCO1)NCC1(COC)CN(C(=O)C(C(C)C)OC)C1 c1(C(=O)NCC(CO)NC(c2cc(F)c(F)c(F)c2F)=O)c(F)cccc1[N+](=O)[O-] Cc1cc(Cl)ccc1NC(=O)C(=O)NCC(O)CNC(=O)C(C)(C)C1CCCC1 S(=O)(=O)(CCC(=O)NCC1CCCCN(C(=O)C(F)=C(C)C2CC2)C1)NC C1(NC(C(=CC2CCCC2)C)=O)CC(O)CN(C(=O)Cc2n[nH]cc2Br)C1 C1(NC(c2csnn2)=O)C2CCN(C(C3(CCO)CC3)=O)CCC12 N1(CC=C)C(=S)NC(c2cnc(C(=O)OCC)s2)C2=C1C(C)(C)NC2=O c1(OCOC)ccc(C(=O)NCCN(C(c2cn(C)c(C)n2)=O)CC)cc1OC c1(-c2n(CCc3ccc(C)cc3)nc(CS(C)(=O)=O)n2)ccc2c(c1)CCCO2 O(NC(=O)C(c1ccc(C)cc1)SC)CC(=O)NC(C#C)CC Cc1[nH]c(C(=O)NCC2CCN(C(c3ccc(C(C)C)s3)=O)C2(C)C)c(C)c1C N1(C(=O)NC(c2ccc(F)cc2)CCC)CCC12CCCC2 Cc1cnc2n1CC(C(=O)NC(C)CC1CN(C(=O)C(C)(C)CCC#N)C1)CC2 Cc1c[nH]c(C(=O)NCC(C)=CC(=O)NC2(c3cccs3)CC2C)c1 NS(=O)(=O)c1ccc(C(N2CCCC2CNC(c2c(F)ccnc2F)=O)=O)s1 C1(C(=O)NC(C(C)(C)NC(C2(C)C(C)C2)=O)C23CC(C2)C3)CCC=CO1 C1(C)(C(=O)NC(c2ccc(N3CCCOC3=O)cc2)C)CC(=O)CCO1 C1(NC(C2(C)CCNC2=O)=O)CN(C(C2CC(O)C2)=O)CC2(CC2)C1 CCCC(C(=O)N1CC(CNC(=O)COCCCC(C)C)(COC)C1)OC Cc1ccc(F)c(-c2ccc(NCc3ccn(-c4ccccc4)n3)cn2)n1 Cc1cc(=NC(=O)C(=O)NC2CC3CCC2N(C(C2CC(F)(CO)C2)=O)C3)[nH]o1 CCCCCCC(F)C(=O)N1CCN(C(=O)C=CCF)C(CC(=O)NC)C1 C(N=c1cc(C)nc(C)[nH]1)C1OCCCN(C(CCCOC)=O)C1 S(=O)(=O)(c1csc(C(=O)OC)c1Cl)NCCC(COC)OC c1(C(=O)Nc2c(OC)ccc(C)c2)cnc2c(C3=CCN(C)CC3)cnn2c1 N1(C(c2c(OC)cc(C)s2)=O)CC(O)CC1(C)C(N1CC(C)OCC1C)=O C1(CCNC(c2cnn(CC)c2Br)=O)CCCN(C(=O)CSC(C)C)CC1 N1(C(C(CC=C)CNC(c2[nH]cc(C)c2C)=O)=O)CCC(C)(O)C(O)C1 Cc1nn2cc[nH]c(=O)c2c1C(=O)NC1CN(C(c2cnc[nH]c2=N)=O)CC1C C1(NC(CC(C)n2cccn2)=O)CC(C(=O)NOCC(O)C(C)(C)C)C12CCC2 Cc1ccc2[nH]c(C(N3CCOC(C(=O)NCC(C)O)C3)=O)cc2c1 c1(C(=O)NC(CNC(c2c(CC)ccc(F)c2)=O)C)cc2sccc2n1C N1(C(C2CCCC2)=O)CCCC(CNCc2cccnc2)C1.c12cccc(c1)S2 c1(CN2CC(NC(c3ncccc3Cl)=O)C(F)(F)C2)cc(Cl)c(O)c(Cl)c1 C(=O)(CC(C)(C)n1cc(CN(C)C)nn1)N1CC(CC)(OC)C1.C1(N)CCNCC1 N1(C(C)C)N=C(C(=O)N2CC3CC2CN3C(c2ccccc2Cl)=O)CCC1=O C(C(C(F)(F)F)OC)C(N1C(Cn2cc(CC(COC)O)nn2)CC1)=O c1(NC(=O)NCC2CCC3(COC3)OC2)cccc2cc(F)ccc12 c1(C(=O)NCCCCNC(c2cccc(C)c2N)=O)ccc2ncc(=O)[nH]c2c1 N1(C(Cc2c(C)cccn2)=O)CCC(NC(c2cc[n+]([O-])cc2)=O)C(F)(F)CC1 c1(-n2cc(C3N(C(=O)NC4CCCS4(=O)=O)CCCC3)nn2)cc(Cl)nc(Cl)c1 Cc1nc(-n2cccc2)sc1C(N1CCC(C2(c3cccc(Cl)n3)CC2)CC1)=O C1(N(C(C=C(CNC(C(C)OCC)=O)C)=O)C)CCOC(C)(C)C1 Cc1cccc(C(=O)NCC(N2CCN(Cc3noc(C(N)=O)n3)CC2)=O)c1F c1(C(N(CCC(N2CC(CC#C)OCC2)=O)CCCO)=O)cccc(O)c1C Cn1ccc2nc(NC(C3CC3C(N3CCCC3c3ccccc3)=O)=O)ncc12 c1(C(=O)NCC2CCN2C(=O)CCc2ncc[nH]2)cc2c(cc1Br)CCN2 c1(SC)ncc(CNCC23C(CN(C(=O)C4CC4)C2)C3)c(O)n1 C(=O)(CCCCCN(C)C(C1CC(OC)C1)=O)N1CC(C#N)(OC)C1 c1(C(=O)NCC2(CNC(=O)C#CC3CC3)CC2)ccc([N+](=O)[O-])cc1Br Cc1cn2cccc(C(=O)NC3CCN(C(C4CC(=O)N(C)C4)=O)C(C)C3)c2n1 c1(SCC)ccccc1CC(=O)NCC1(NC(c2cnn(C3CC3)c2)=O)CC1 N1(C(C(=O)NCC(C)O)C)CCCOC(CNC(=O)CC(C)(C)C)C1 C(C(CC(F)(F)F)NC(c1c[n+]([O-])c(C)cn1)=O)NC(C=Cc1ccc(C)s1)=O CCCCCCC(=O)NCCN(C(=O)Cc1scnc1-c1cccs1)CCOC NS(=O)(=O)c1ccc(C(=O)NCC(CO)NC(C2CNC(=O)N2)=O)c(Cl)c1 N1(C(C23OCC(C)(C2)C3)=O)C2CCCC1CN(C(C1CC13CCC3)=O)CC2 c1(CNC(c2ocnc2C(C)C)=O)cc(C(=O)NCCc2cc[nH]n2)cs1 C(=O)(CC(COC)NC(=O)Cc1ccc(F)cc1)N(CCC)CCO C1(CN(C(=O)C(F)C2CCC2)C)CN(C(c2ccon2)=O)CCO1 C12(CC)CCC(C(N3CC(NC(=O)C(F)(F)c4nccs4)C(F)C3)=O)(CO1)C2 C1(CC(N2CC(CC(C(=O)N(C3CCCC3)C)F)C2)=O)CC(C)(C)CO1 c1(C(c2nnnn2CC2CCOC2)NC2(CC=C)CC2)cc2ccccc2o1 N1(C(CC(C)(C)N(C)C(C2CC3CCC(C2)O3)=O)=O)CCC2(COC(=O)N2)C1 CC1=C(C(=O)NC2CCN(C(=O)C=Cc3nccs3)CC2F)CCS1(=O)=O C1(C(N2CCC(N(C(c3c(C)nc[nH]3)=O)C)CC2)=O)CC(C)(C)CN1C N1(C(C(=O)Nc2c(C)cc(F)cc2)C)CC2C3CCC(CC3)C2C1 c1(C(N(C2CCN(C(C3SCCS3)=O)C2)CC)=O)ncccc1N C1(C(N(C2CCN(C(c3cccc(OC)c3F)=O)C2)C)=O)CCCCC12CCC2 c1(CCC)ncc(NC(C(=O)N(CCCN(CCC)C(C)C)C)c2ccco2)s1 N1(CC2CC(NC(=O)Cc3cn[nH]c3)OC2)CCCC1CC1(OCC(=O)OC)CC1 CC1=C(C)CC(C(=O)NC2CC(CCNC(=O)CC3CCSCC3)C2)CC1 c1(CN(OC)C(=O)c2nc(C)n(C)n2)cc(C)ccc1C N1(C(Cc2c(C)nsc2)=O)CCN(C(C2CCOC2C)=O)CC1CC(F)(F)F c1(COC)csc(C(=O)NCC2CCN(C(C3COCC3OC)=O)C2)c1.C1CC1 N1(C(c2ccn(CCC)n2)=O)CC(C(=O)NC(c2cscn2)CO)C(C2CC2)C1 C=CC(F)(F)C(=O)N(C(C)(C)CC(=O)N(C1CCCCC1OC)C)C CC(C)C(C)C(=O)NC(C)CCC(=O)NC1(CCF)CC1 C1(CN(C(=O)CCc2ccoc2)C2CC2)CCCCN1C(=O)C=CC=C(Cl)Cl N1(C(c2n(C)cc(F)c2)=O)CCCC(O)(CNC(c2cccc(F)c2F)=O)C1 C1(C(N2CC3(CN(C(CCCOCC=C)=O)C3)C2)=O)COc2ccccc2O1 c1(OC)ccc(S(=O)(=O)NCC(=O)NC2CCC2)cc1.C12CCCC1N2 c1(C(=O)NC2C(CNC(C(C=C)O)=O)C2)ccc(Br)c2c1OCCC2 CS(=O)(=O)CC(=O)N1CCN(CCNC(c2ccc(C(N)=O)[nH]2)=O)CC1 c1(N(CCCC=C)C)nc(=NCC2CCCS2)[nH]c2c(C)nn(C)c12 C1(NC(CC2(C#C)CCC2)=O)CN(C(c2cc(Cl)ncc2OC)=O)C(C)(C)C1 CC(F)(CNC(=O)C(=C1CCCCC1)F)CNC(C1OCCC1C(F)(F)F)=O c1(C(=O)NCC(CCNC(C(C=CC)O)=O)O)cc(C)cc([N+](=O)[O-])c1 CCC(C)(C(=O)NCC(C)CN(C)C(c1ccncc1-n1cccn1)=O)OC C(=O)(CC1=NNC(=O)C1)NC(C)CCNC(c1ccc(CN2CCOCC2)o1)=O CC(N=c1cc(C(F)(F)F)nc(-c2ccccc2)[nH]1)c1c(F)cccc1F CCC1=C(C(=O)NCC2CC(O)CN2C(=O)CC(COC)COC)CCCO1 CC1C(NC(=O)C(F)C(F)(F)F)CC2CCC1N2C(=O)CC1C=CS(=O)(=O)C1 c1(C(=O)NC(C)C(C)NC(c2cc(Cl)ccc2Cl)=O)ccc2sncc2c1 C1(C(N(C(C)CNC(c2c[nH]c(=S)cn2)=O)C)=O)CCOCC1(C)C C1(NC(CN(C2C(C)C2)C)=O)(CF)CCN(C(C2CC2(C)C)=O)C1 N1(C(c2cnco2)=O)CC2=C(C1)CN(C(c1ccnn1C1CC1(F)F)=O)C2 c1(CCCCC)ccc(NC(C2CCC(NC(=O)CN3CC=CC3)CC2)=O)cc1 C1(C(N2CCC(C)CC2)=O)CC2CCN(Cc3cccc(=O)n3O)CC12 N1(C(C2C(n3cc(CNC=O)nn3)COC2)=O)CC2COCC(C2)C1 CCC(CC(=O)NC1CC(F)(CNC(C2CCCC(C)(C)C2)=O)C1)C(C)(C)C N1(C(C=COCC)=O)CC2CCC(C1CO)N2C(c1cc(OC2CC2)ccn1)=O c1(NC(C2(C)CCCC2CNC(C=CC(CC)C)=O)=O)cc(CO)cc(F)c1 C1(NC(C(CCC)OC)=O)CN(C(c2cccc3c[nH]nc23)=O)C2(CCC2)C1 C1(NC2CCC(S3=CC(C4CC4)=N3)CC2)CC2CCC1C2 C1(N(C(C(N(C(COC(CC)CC)=O)C)C2CC2)=O)CC)CCNC1=O CC1CCN(C(=O)C(C)(C)c2cncnc2)CC1NC(=O)Cc1nccs1 C(=O)(CCCCCc1ccccc1)NC(CN(C(c1n(C(C)C)ncn1)=O)C)C C(C(=O)NC1CCCC1C(C)C)(C(C)O)NC(c1c(CC)cno1)=O C1(CC(N2CC(CCNC(=O)Cn3nnc(C)n3)C(C)C2)=O)(OC)CCOCC1 C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CC=CC(NC(CCc2onc(C)n2)=O)C1 Oc1cccc2c1CN(N1CCCC(Oc3ccccc3)C1)CCO2 C1(C(=O)NCC(COC)NC(C23COCC2C3)=O)CCCC(CF)C1 c1(C(=O)NCC2CC(NC(CC(=C)C)=O)C2)c(C)nnn1C N1(C(CC(C)C)=O)CCC2CN(C(C3CCN(c4ccc(Cl)cc4)C3=O)=O)C2C1 C(=O)(C1Cc2ccccc21)NCCCC1N(C(c2c(C)cccc2)=O)CCCC1 Cc1noc(CCCNC(=O)C=CC(C)NC(c2cc(Cl)c[nH]2)=O)n1 c1(C(N2CCN(C(=O)Cc3cnoc3)CC2CF)=O)sc2sccc2c1Cl CC1(CNC(C2CCN2CC2C3COCC23)=O)CCOCC1 C1(NC(c2cccc(C)c2Cl)=O)CCN(C(=O)C=Cc2cccs2)CC1(C)C CN1CCN(C(=O)C=Cc2cncn2C)C(C(=O)NCc2cccc(CO)n2)C1 c1(C(=O)NCC(CNC(Cc2ccc(OC)cn2)=O)O)cccc2c1nnn2C N1(C(CC2C(C)C2)=O)CCCC(C(C)(O)CNC(=O)C=C2CCOCC2)C1 CCC(C(C)(C)O)NC(C1(C)CN(C(c2sccc2C#N)=O)C1)=O N1(C(c2cc(C)nnc2O)=O)CCC2CN(C(=O)CCC3CCCOC3)CC12 c1(CC(C(=O)OC)COC(c2ccc(OCC3CC3)cc2)=O)ccc(C)cc1F C(=O)(C(Cc1cc[nH]n1)NC(c1ncccn1)=O)N(CC#C)C c1(C(=O)NC2CC3CN(C(CN(C)CCO)=O)C2C3)cc2cccn2c(O)n1 N1(c2n(CCOCC=C)c(C(=O)OC)nn2)Cc2ccccc2OCC1C(F)F CCCC(F)C(=O)NC1(C)CCC(OCCNC(=O)Cn2ccnc2C)C1 C1(c2scc(OCC)n2)CN(C(=O)CCCOC)CCN1C(=O)C1=NOC(C)C1 Cn1c(=O)nc(O)c2cc(C(=O)OCc3ccc[nH]3)cnc12 C1(OCC)CC(CC(=O)N(C)CCOC)C1.C12(CC1)C(=O)N2 N1(C(C(C)CF)=O)CCC2(CCC2)C(NC(C2C=CC=CC=C2)=O)C1 c1(OC)cccc(CCC(=O)NC2CC2NC(=O)C=Cc2cn(C)cn2)c1F C1(C(CO)NC(=O)CC(Cl)Cl)CCN(C(C2CC2F)=O)CC1 C1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCSCCOC)CCN(C)C1=O c1(C(N2CCC(N(C(=O)C(O)C(C)CC)CC)C2)=O)ccc2c(c1)CCOC2 C(=O)(CCCCCCn1cc(CN)nn1)NCCC(C)OCCOC C(CC(=O)NCc1ccccc1CO)(C(F)F)NC(=O)CC12COC(C1)C2 c1(NCC2C(NC(c3c(OCC)cccc3)=O)CCC2)ncnc2c1CCO2 CC1CCC(C)(CS(=O)C(C)Cc2ccc(Cl)s2)C1 N1(C(CC=C)=O)CCC2CN(C(c3c4c(nn3C)CCOC4)=O)CC2CC1 CC1OC2(C)CC1(NC(=O)CC1CCCN(C(=O)C=CC3CCCC3)CC1)C2 C1(C(N(CCC(=O)NC(C)C(C)CO)CC=C)=O)CC2(CSC2)C1 C(C)(CN=c1[nH]nc(-c2ccc(C(F)(F)F)cc2)o1)N(C(C)=O)C c1(CC)cc(C(N2CCC(NC(=O)CCNC(=O)COC)C(O)C2)=O)ccc1O C=C(CNC(CCC(C)C)=O)CCNC(c1cnoc1-c1ccc(C)o1)=O C1(C)(NC(CCc2scc(C)n2)=O)CCN(C(C2CCC(C(N)=O)CC2)=O)C1 c1(C(N(CC(C)(C)NC(c2n(COC)ncc2)=O)C)=O)cc(C(C)C)cnc1O c1(-c2nn(C(C=C)C)c(-c3cc(-c4cccs4)[nH]n3)n2)ccc(F)c(Cl)c1 C1(C2(O)CCOC2)(NC(=O)CC2CN(Cc3ccccc3)CCO2)CC1 C1(=O)CCC(F)(F)CO1.c1(C2C(C(=O)OC)CCC2)ccc(Cl)cc1 N1(C(=O)NCCCC(=O)NC)CCOCC12COC2 c1(C(=O)OCC)ccccc1C(=O)NC1(CNC(CC2C(C(=O)NC)C2)=O)CC1 C1(C2CN(C(C3(C)CCN(C)C3)=O)C2)(NC(C2C(C#C)C2)=O)CC1 C1(O)(CNC(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC1 C1(CN(C(CCNC(COC)=O)=O)C)CCCCN1C(c1cc(F)c[nH]1)=O C1(C(=O)NCCN(CCC)C(=O)CN2CCC(C)(O)C2)OCCCC1(C)C N1(C(c2cc(C)cc(C)n2)=O)CC(NC(=O)C(C)(C)CO)CC12CCCOC2 C1(C(=O)NC2C(C)(C(C)C)C2)CCN(C(=O)C(=O)NC2CC2)C1C(C)C CS(=O)(=O)C(C(=O)NCC#CCNC(C12CC(CN1C1CC1)C2)=O)C1CC1 c1(OC)cccc(C(C)NC(=O)CCCn2cc(CCN3CCOCC3)nn2)n1 C(=O)(CN=c1cc[nH]cc1)N1CCC(C(N(C)CCc2nccs2)=O)C12CCC2 C1(C(=O)NC(C(=O)OCC)C)CCN(C(C2CC23CCC3)=O)C1(C)C N1(C(CCCOC)=O)CCC2(CCCC2NC(C2CC(C(C)(C)C)=NO2)=O)CC1 c1(C(=O)NC(CC)CNC(c2ccc(=O)n(C)c2)=O)cc(F)cc2cccnc12 C(=O)(C(C)(C)CC(=O)N(CCNC(c1c(Cl)c(C)nn1C)=O)C1CC1)OCC c1(CC(=O)NC2CCC(CNC(CCNC(N)=O)=O)C2)cc2c([nH]1)CCCC2=O c1(C(=O)NC2CCCN(C(CCCNC(C)=O)=O)CC2)cncc2ncn(C)c12 N1(C(C=CC(CC)=CC)=O)CCN(C(c2cnc(NC)cn2)=O)CC1C(C)(C)C C1(NC(C(CC(C)C)O)=O)CC12CCN(C(=O)CC1(C)CCCCC1)CC2 C1(NC(C(CC=C)C)=O)CCCCC12CCCN(C(=O)CC1CCCC1(F)F)C2 N1(C(C(C)C#N)=O)CCCCC(CNC(c2ccc(C#N)s2)=O)C1 c1(C(=O)NC(C)CNC(C2OCCC2C)=O)ccc(F)c2ccsc12 CC(C)C(C(C)NC(c1scnc1Cl)=O)NC(=O)CN(CC(C)(C)C)C C1(CCNC(C(C)CN(C)C)=O)CSCCN1C(=O)C=Cc1cc[nH]c1 c1(OCC)ncc(C(=O)NCC2(F)CCCN(C(=O)CCC(C)O)C2)cc1Cl C1(CC(=O)NCC2(C)CCCN2C(c2cc(C3CC3)on2)=O)CC(O)C12CCC2 N1(C(C(COC)C)=O)CCCC(C)(C(=O)N(CCCO)C2CCC2)C1 c1(C(=O)NC(C(C)NC(c2c(COC)cco2)=O)C)c(C)cc(C)cc1N c1(N2C(CNC(C3CCOC3)=O)CC3(CC3)C2)ncnc2ccc(I)cc12 C1(CNC(C(C)=CC)=O)CCCN(C(c2c[nH]cc(Br)c2=N)=O)CC1 N1(C(CCCOCC)=O)CCC(O)C1C(N1CCC(N2CC(O)C2)C1)=O N1(C(CC(C)(C)NC(C(CC#C)C2CC2)=O)=O)CCC12CCN(C)C2 C(=O)(C(C)(C)CC(F)F)N1CC(C)C(NC(=O)C(C)c2ccon2)C1 C(=O)(CN1C(=O)C(F)(F)Oc2ccccc21)NC1CN(C(COC)=O)C2C1C2 C(=O)(C1CCc2cc(F)ccc21)NC(CC)CNC(c1cc(C(F)F)on1)=O C1(C(C)C)C(NC(=O)CCCCN(C)C)CCN1C(=O)CCCn1cncn1 CC1CCN(CC(=O)N(C)CCN2CCN(C(=O)C(C)(C)C3CCC3)CC2)CC1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)cnn2C(C)C)=O)cccc(CC)c1 N1(C(CC2CC(CC)C2)=O)CCC(C(=O)OC)C1Cc1ccc(C(=O)OC)s1 n1(CC)cc(Cl)c(C(=O)N(CC(CO)(CO)NC(C2CC2(F)F)=O)C)n1 c1(NC(C(C)Cn2cccn2)=O)cccc(CNC(C2COCC2(C)C)=O)c1 C1(C(=O)NCC2(NC(c3nnn(-c4ccccc4)n3)=O)CCC2)C2CC2C2CC12 c1(SC)ccc(C(=O)NCC(C)(C)NC(=O)NC(C(=O)NC2CC2)C(C)C)cc1F CCN=C(NCc1cccc(NCCO)c1)NCC(C)(C)C(=O)OC(C)(C)C O=C(CCC1=CCCCC1)NC1CCN(C(c2ccnc(OCF)c2)=O)C1 c1(C(=O)NCC2N(C(c3c(COC)cco3)=O)CCC2C)c(C)cc(O)nc1C N1(C(C(n2cc(Br)cn2)C)=O)CCC2(CCC(NC(=O)CC3CC3)C2)CC1 Cc1ccc(C(=O)NCCC2(O)CCCN(C(=O)C(C)C3(O)CCC3)C2)cc1N N1(Cc2n(CC)ncc2)CCCC(CO)(NC(c2ccc(Cl)nc2OC)=O)C1 CCC(CC)CCC(=O)N(C)CC1CCCN1C(C1CC2(CCO1)CC2)=O C1(NC(CCSCC)=O)CC2CN(C(c3cnc(Cl)s3)=O)CCN2C1=O N1(C(c2ccc(OC)nc2Cl)=O)CCN(C(C2OCCC2C)=O)C(C)C1C N1(C(c2cscc2F)=O)CCC2CN(C(=O)CSc3ccc([N+](=O)[O-])cc3)C2C1 c1(C(=O)NCC23CCC(CN2C(c2ccnnc2)=O)C3)ccn2nncc2c1 c1(-c2cc(C)[nH]n2)ccc2c(C(N3CCNC(=O)CC3)=O)c[nH]c2c1.C(C)(C)(C)N c1(CCNC(C(C)OC2CCN(C(=O)CC(O)C3CC3)C2)=O)ccc(F)c(F)c1 CC(CO)(CO)NC(C1C(NC(c2nsnc2O)=O)C1(C)C)=O C(=O)(C(C)CC(=O)OC)N1CCC(CC(=O)NCC2(C(=O)OC)CCC2)C1 C1(NC(CN(CCC)C)=O)CCCCC1C(=O)NC1CC1C1CC1C C1(C(N2CCC(NC(C(OC)OC)=O)CC2C)=O)CC2(C1)CC1(CC1)C2 c1(C(C)OC)nc(CC(N2CC(O)(CNC(=O)CSc3n[nH]c(C)n3)C2)=O)cs1 C1(CC)CN(C(=O)CN(CC(C)C)C)CCN1C(=O)CNC(c1ccccc1)=O C(N=c1[nH]c(=NCc2cccc(Cl)c2F)[nH]c2c1CCCC2)c1c(C)ncs1 C1(C(=O)NCCC2CCCN(C(c3c[nH]nc3C(F)F)=O)C2)CCCCC(=O)N1 c1(C(=O)NC2CN(C(Cn3c(C)cc([N+](=O)[O-])n3)=O)C2)nccc2c1NCCC2 N1(C(C(OCC)OCC)=O)CC2CCCC2C1C(=O)NCc1[nH]nc(CC)c1C c1(OCC)ncc(C(=O)NCC2CCCCN2C(=O)CC(C)(C)SC)cc1Cl c1(C(=O)NC2CC(NC(C(CCC#C)O)=O)C2)cc(F)cc2nn(C)cc12 C1(NC(Cc2c(C)n[nH]c2C)=O)CN(C(=O)CC(C)C(C)(C)C)CC(F)(F)C1 c1(Cn2ncc(C(=O)NCC3(NC(=O)CO)CC3)c2)ccc(F)cc1F C=CC(C)(CCOC)C(=O)NCC1CCCCN1C(=O)Cc1cccnc1 C(=O)(C(C)C(F)(F)C(F)F)N1CCC(N(C(C2CCC(OCC)CC2)=O)CC)CC1 c1(CC(=O)NC(n2c(C)cc(C(=O)O)n2)(C)C)cc2ccccc2o1 Cc1nc(N2CCC(NC(C3CCCC3C(C)O)=O)C2)c(C)c(C)n1 c1(Nc2n(C)ncc2C2CC2)cn2c(nc1=O)SCC2.C12(CC1)CNC(=O)NC2 C(=O)(C1CCc2cccc(O)c21)N1CC(NC(C(c2cnccn2)C)=O)C(C)C1 C1(CC)CN(C(=O)COC2CC=CC2)CC1C(N1CC(O)(CO)C1)=O c1(C(=O)NCC2(CNC(CC(CC)OC)=O)CCCCC2)cc(F)ccc1OC C1(F)(C(N2CC3C(NCc4ccc(C)cc4C)C3C2)=O)CCCCC1(F)F c1(C(=O)NCC2(NC(C(C)OCCOCC)=O)CCCC2)nccc2occc12 c1(C(N(CCNC(C(COC)N(C)C)=O)C(C)C)=O)ccc(F)c2cccnc12 N1(C(CCCOC)=O)CC(N(C(=O)CC(C(F)F)c2ccccc2F)C)C(F)C1 c1(OCC)c(C(=O)NC2CC(C(=O)Nc3cc(F)ccc3I)C2)cccc1F C1(CNC(c2cccc(SCCOC)c2)=O)CCN(CC2CCC2C)CC1 C(=O)(CCS(C)(=O)=O)NC1CCCC(CNC(c2n(C)nc(C(F)(F)F)c2)=O)C1 C1(C(N2C(C(=O)NC(C3CCOC3)C#C)CC2C)=O)CC(=O)NC(=O)C1 CC1CC(NCC=CCCF)CN1C(=O)C(F)=C1CCC1 C(C(C)(C)CS(=O)(=O)CC)NC(c1ncc(Cl)cc1F)c1n(CC)nnn1 N1(C(C2CC(=C)C2)=O)CC(NC(=O)CCn2ccnc2)Cc2ccccc21 C(=O)(CC(C)(C)C(C)(F)F)NC(C1(O)CN(C(=O)Cn2cc(Br)cn2)C1)C Fc1cc(CNCC2CCCCCC2(F)F)c2c(c1)CCO2 CC(C)C1=NOC(C(N2CCCC2CN(C)C(c2conc2C2CC2)=O)=O)C1 c1(NC(CCCC=C)C2CC2)ncc(S(=O)(=O)NCC2(CC)CCOC2)cc1Cl C(=O)(C#CC1CCOCC1)N1C(CN(C(C2C=CCCC2)=O)CC)CCC1 c1(-c2cnc(CN(C(C(=O)NC)CC(C)C)C)nc2)cccc(C#N)c1C C1(F)(C(=O)N(C2CC2C(=O)O)CC2CCOC2)CCCCC1 C(=O)(C1=C(Cl)CCCC1)N(C(C)CCNC(C1CC1[N+](=O)[O-])=O)C N1(C(CCNC(C2CC(O)(CC#C)C2)=O)=O)CCCCC1C1(O)CC1 Cc1cc(C(=O)NC2CCCC2CC(=O)NC(C)C2CC2)cc(O)n1 c1(C(N2CC(OC)(CNC(=O)C(c3ccccc3)F)C2)=O)cc2c(ccn2C)[nH]1 N1(C(=O)C=C2CCCCC2)CCC2(CC1)CN(C(C13COCC1C3)=O)C2 C1(NC(CN2CC=C(C)CC2)=O)CCCN(C(c2cccc(Cl)c2)=O)C1C CCC(O)C(C)(C)C(=O)N1CCCC(N(C(=O)Cc2cnc(C)s2)C)CC1 C(CCCC(C(=O)NC(C)C(=O)OC)N1CC2(CC=CC2)C1c1ccccc1)OC C#Cc1cnn(C)c1C(=O)N(C)CC1CCCN(C(C2CCN(CC)C2)=O)C1 O=C(C1=COc2ccccc2O1)NC1(CCCNC(c2ncccc2F)=O)CC1 N1(C(C2CCCN(C(C=CCC)=O)C2)=O)CCOC(C2CC2)CC1 c1(C(N(CCCN(C(C(C)OCC(F)(F)F)=O)C)C)=O)coc(COC)c1 c1(NC(C2CC23CN(Cc2cccc(Cl)c2)C3)=O)nccc2cccnc12 Cc1cccc(C)c1C1(C(=O)NCC(C(C)C)NC(=O)C(O)C2CC2)CCC1 N1(C(c2cc(CC)nn2C)=O)CCN(C(=O)CCC2(C)CC2)C2CS(=O)(=O)CC12 C1(C(=O)NC(CCC)C)CCCC12CCN(C(=O)Cc1cccn1C)C2 c1(C(N2C(C)CC(NC(=O)CN3CCC(C)(O)C3)CC2)=O)cc2c[nH]cnc-2n1 N1(C(C(CC=C)N(C)C)=O)CC2(C(=O)NCc3ccc(OC)c(F)c3)CC1CO2 N1(C(c2cncc(OC)c2)=O)CC2CCN(C(C3CC3(F)F)=O)CCC2C1 c1(N2CCC(CN(C(C(C)Sc3ccccn3)=O)C)CC2)ncnc2c1COC2 Cc1cc(C(N2CC(NC(=O)C3=CCSC3)CC23CCCC3)=O)cc2ccoc12 C=C(C)C1CN(C(=O)CCN(C(C2CC2=C)=O)CC)CCO1 N1(C(c2n(CCOC)ncc2)=O)CCCC(NC(c2cncn(C)c2=O)=O)C1C C12(C(N3CCN(CC(=O)NC(C4CCSC4)C)CC3)=O)CCN(CC1)CC2 c1(NC(C2OCCN(C(C(C)Oc3ccccc3)=O)C2)=O)ncc(F)cc1Cl c1(C(CNC(C(C)C2CCCC2)=O)(F)F)nnc2ccccn12 C=CC1(CC(=O)NCC=CCNC(c2c(C)coc2C)=O)CCCCC1 CCCCCC(F)C(=O)N1CC(=O)CC1C(=O)NCC(C)N(CC)CC c1(N(C(C(CC2CCCC2)NC(C(C2CC2)OC)=O)=O)C)cc(C)cc(C)c1 C(CNC(=O)C=C(Cl)Cl)(C(C)C(C)C)NC(C(C)(C)OC(C)C)=O C1(C(=O)NCC2N(C(c3n[nH]c(C)c3Cl)=O)C3C(C2)C3)CCC(C)(C)CC1 c1(NCC2(NC(C3CC3c3ccc(F)cc3)=O)CCC2)ccc2nccn2c1 C1(CNC(c2nc(CC(C)C)sc2)=O)CC(NC(c2cc[nH]n2)=O)C1(C)C C1(C(N(CCN(C(C(C)Oc2ccccc2Cl)=O)C)C)=O)Cc2ccccc2S1 c1(OC)cc(Br)c(NC(C2CCN2C(c2ccc(C(F)(F)F)cn2)=O)=O)cc1C CC(O)C(C)C(=O)N(C)CCOCCCN(C(=O)C(C)(C)c1ccns1)C C1(NC(c2n(CC)ncc2)=O)CC(C)N(C(=O)CCCOc2ccccc2Cl)C1 C1(C(N2C(C)C(NC(c3cc(Cl)c[nH]3)=O)CC2)=O)CCc2ccccc2N1 C=CCCCCCC(=O)N(C(CNC(=O)CC1C=CS(=O)(=O)C1)C1CC1)C C1(C(N)=O)(CNC(C(CC)OC)=O)CCCN(C(=O)CCC2CCCC2)C1 N1(C(C2C(=C)C2)=O)CC2CCC1C1CN(C(=O)C(CC)CC)CC21 N1(C(C(C)C(C)O)=O)CC2(CCN(C(C3SCCS3)=O)CC2)CC1C C1(NC(C2C(COC)C2)=O)CC2CN(C(c3cnc4n3CCC4)=O)CC12 N(C1CC2(CN(C(=O)Cc3cccnc3)C2)n2ccnc21)C(CCC(C)(C)F)=O CC1=C(C(=O)NC2CC2NC(=O)C=Cc2cscn2)Cn2nnnc2N1C N1(C(c2c(Cl)ccc(N)c2)=O)CC2CC1CN(C(=O)CCn1cnccc1=O)C2 C1(CN(C)C(c2nccnc2C(N)=O)=O)CCCCN1C(c1cnc(O)o1)=O C1(C(=O)NC2(C)CN(C(C(C(C)C)SC)=O)C2)CC(C)CC(C)C1 c1(C2(C(N(CC)CC)=O)CC2)ccc(F)cn1.C1(=O)CC(=O)NCCCCCN1 c1(OCCC)ccc(C)cc1-c1cnc(NC(=O)Cc2ccc(Br)cn2)c(C)c1 c1(C(=O)OCC2CCC(F)(F)C2)ccc2c(n1)OCCO2 c1(NC(=O)NC(COC)C)nc2ccc(OC)cc2c(=NCCC(C)(C)F)[nH]1 C1(CNC(=O)CCc2cncs2)CCCN1C(C1(C(F)F)CCCO1)=O CCC(C)(C(=O)NCC(C)(C)NC(=O)C(C)(c1ccccc1)OC(C)C)C(F)F C1(C(=O)NC2C(NC(CCSCCC)=O)COC2)CN2CCN1C(C)C2 c1(C2C(NC(=O)OC)CCC2)ccc(OC(=O)C(C)(O)Cc2ccccc2)cc1 C(=O)(C(C)CC(F)(F)F)NCC1(O)CCN(C(COC2(C#C)COC2)=O)C1 CCCC(CC)C(=O)N1CCN(C(=O)CCN2CCSC(C)(C)C2)CC1C(C)C C1(CCC)CN(C(CC(F)F)=O)CCN1C(=O)C(c1ccc(C(C)C)c(Cl)c1)=O Cc1ccc(S(=O)(=O)N2CC=CC2C(=O)Nc2cncnc2I)cc1C C1(C(N2CC(OCCOC)C2)=O)CC(C)CN(C(=O)C(C(C)C)NC=O)C1 Cc1nc(N2CCC(C(C)C#N)CC2)cc(-c2ccccc2)n1 C(CN=c1nn[nH]n1C)C1CCN(C(c2c(C)snc2)=O)C1 C1(CNC(Cc2cc(C)no2)=O)COCCN1C(=O)C(O)CN(C)C C1(NC(CCCC)=O)CCN(C(=O)Cc2ccnc(F)c2)C1(C)C N1(C(CC2(CNC(c3cc(COC)[nH]n3)=O)CC2)=O)CCC2CCNC(=O)C12 CC1CCN(C(c2cocn2)=O)C(C)C1NC(C1CS(=O)(=O)CC(=O)N1)=O c1(CCC(=O)NC2CCCC2NC(C2CCCC2O)=O)cnc2n1CCCC2 C(=O)(C(C)CCC(C)(C)C)N(C)CC1CCCN(C(=O)C(CO)C(C)(C)C)C1 N1(C(=O)NCC2(C#N)CCCC2)CCN2C3CCC(C3)C2C1 N1(C(Cc2ccc(C)o2)=O)CCC(F)(C(=O)NC(CC)C(C)CN(C)C)CC1 C(=O)(CCCCN1CCCCC1)NC(C)(C)CCNC(C1(C2CCCO2)CC1)=O CC1(C)CCC(C2CCCCN2c2ccnc(NC3CC4CCC3C4)n2)C1 N1(C(C23C(C)OC(C)(C2)C3)=O)CCC2(CC1)CCN(C(C1CC3(CC3)CO1)=O)CC2 C1(CNC(c2cccc(C)c2)=O)CC2(CO1)CN(C(=O)C(c1cnn(C)c1)=O)C2 C1(CNC(=O)CN2CCSCC2)CC(F)CN1C(=O)COC.C1(O)CCCC1 C1(C(=O)NC2(C(=O)OC)CCOC2)(NC(C(COC)C)=O)CCN(C)C1 c1(CN2C(CCCNC(C(C(C)C)SC)=O)CCC2)cn(C)c2cccc(C)c12 c1(C(C(=O)N(CC(CC)NC(c2sccc2SC)=O)C)O)cncn1C C1(C)(CNC(C2CC(OCC)C2)=O)CCCN(C(C2(C)CCC3CC3C2)=O)C1 C1(C(=O)NCCCn2cnnn2)CCC(O)CN1C(=O)C1CC1 c1(C2N(C(c3c(CC)ccs3)C(=O)NC3CCC3)CC2)ccc(N(C)C)cc1 C1(CNC(c2cc(Cl)n[nH]2)=O)CCN(C(=O)C(O)c2ccsc2)CC1 C1(NC(C=C(C)c2ccsc2)=O)COCCN(C(=O)Cc2ccnc(O)c2)C1 N#CCS(=O)(=O)c1ccc(C(N2CCN(C(c3nc(Cl)cs3)=O)CC2)=O)cc1 Cc1ncccc1-c1nc(CN2CCCC2)no1.c12ccccc1N2 CC(O)C(C)(C)C(=O)NC1CCCC(NC(=O)COc2cc(CO)ccc2Cl)C1 C1(C(N(C)Cc2ccnn2C2CCCCC2)=O)CC12CCC(F)(F)CC2 C1(C(=O)NC(C#C)=O)CCCCN(S(C)(=O)=O)C1 c1(C(=O)NCC(C)CNC(=O)CCCCC(F)F)cc(P(C)(C)=O)ccn1 CC(C)C(F)(CNC(=O)CCC(C)N(C)C)C(=O)NCCCn1cncn1 c1(C(C(=O)OCC)N(C)C2CC2)c2c(nn1C)CCC2.C12CCC(CC1)C(=O)N2 N1(C(c2[nH]cc(C(N)=O)c2)=O)CC2CC(NC(=O)Cc3cnns3)C(C2)C1 C(=O)(CC(C)CC(C)(C)C)N1C(NCc2ccc(C(C)C)cc2)COCC1 C1(C)(C(=O)NCC(CN(C)C(c2c[nH]cc(F)c2=O)=O)O)CCCCNC1=O c1(C(=O)NCCC(=C)CNC(C2CCCCN2C)=O)cncc(N)n1 c1(CC)nncn1NC(=O)C1C2CN1C2.c1(C(=O)OC)nnccc1C C(=O)(CC(O)CC(C)(C)C)N1CC(SC)C(NC(=O)CCc2cncs2)C1 C1(N(C(C(C)CC(F)F)=O)C)CC2CCC(C1)N2C(c1ccc(Cl)[nH]1)=O C(=O)(C(O)C(C)(C)C)NCC1(C(N)=O)CN(C(=O)CC23CC(C2)C3)C1 C1(CN2CC(=O)N(Cc3c(OC)ccc(Cl)c3)C2=O)CCC2(CCOCC2)O1 C(C1C(C)C1(Cl)Cl)=CC(=O)NCCN(CCC)C(c1ccc(-c2ccco2)s1)=O C1(N(C(C2C(NC(COCCCCC)=O)CC2)=O)CC)C(=O)OCC1(C)C C=C(Cl)C(C)(C)C(=O)N1C2CCC1C(CNC(=O)CNc1ccccc1Cl)C2 CCCC(CC)C(=O)NC1CC(CCNC(c2c(C)cnn2C)=O)C1 c1(CNC(C2CCN(Cc3ccc(Cl)s3)CC2)=O)cccc(Cl)c1F C1(CNC(C2(C)CC(NC(C3CC=C(C)CC3)=O)C2)=O)CC(=O)N(C)C1=O C1(C(C)(C)C)CCC1(c1nnnn1C1CCOCC1)NCCc1ccsc1Cl N#Cc1cc(F)c(NC(C2CCCN2Cc2cc(-c3ccco3)no2)=O)cc1Cl c1(C(=O)NC2C(CNC(C(C)C)=O)CCC2)cc2scc(Br)c2[nH]1 C(=O)(CC1(C)CCc2ccccc21)NCCCC(C)NC(C1(C)CC1)=O N1(C(C(CCC)N(C)C)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 N1(CCOC)CC(C(=O)NC2(C)CC(NC(=O)C=Cc3ccccc3)C2)CC1=O c1(C(=O)NCCOC(CNC(C(CC)N(C)C)=O)(C)C)ncccc1F Cc1cc(C(N2CCN(c3ccncc3Cl)CC2)C(=O)NCS(N)(=O)=O)sc1Cl C=CCC(C(=O)NCCN(C(=O)C(C)n1cncn1)C1CC1)C(C)C N1(c2cc(C(=O)OC)ncn2)CCCC(NC(=O)Cc2cc(C)no2)C1C C(C(=O)N1CCC(C(C)NC(C2(c3ccccc3F)CCC2)=O)C1)(C(C)C)OC C1(CNC(=O)NCCCCC(OC)OC)C2Cc3c(Br)cccc3C12 N1(C(C(CCCC)NC(C23CC2CNC3=O)=O)=O)CC2CCCC(C1)N2C C1(NC(=O)Cc2cncnc2)CCCCC1CC(N1CC(O)(CN(C)C)C1)=O CC1(CNC(=O)Cc2cccnc2)CCCN(C(C2(F)CCCCC2)=O)C1 C1(CC(=O)NCC2OCC(C)(C)C2)CCN(C(c2cnnn2C2CC2)=O)C1(C)C N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCN(C(C3(O)CCSCC3)=O)C2)C1 C(c1cn(C)cn1)=CC(=O)N(C(CC)CNC(C1CC1Br)=O)CC c1(C(N2CCC(C)(CNC(c3scc(OC)c3)=O)C2)=O)cn(C)c(C)cc1=O N12CCC(CC1)C2=O.c1(C(=O)O)ccc(Cn2cc(C3(O)CCC3)nn2)s1 c1(CC(=O)NCC2N(C(C#CC(C)C)=O)CCC2C)oc2ccccc2c1CO C(c1cccnc1)=CCNC(C1CC(NC(C2CC(COC)C2)=O)C1)=O Nc1nc(Br)ccc1C(=O)NC1CC(F)CN(C(=O)Cn2ncnn2)C1 C1(NC(c2c(Cl)ncc(C)c2)=O)CCN(C(c2c[nH]c(=N)s2)=O)C12CCCC2 c1(C(=O)NCCC(C)NC(C2CN3CCN2C(C)C3)=O)ncnc2c1CCC2 Cc1cccc(C(O)C(=O)NC2CCCCN(C(c3cc(N)ccn3)=O)C2)c1F c1(CN(C2CCC(CC)CC2)C)nccc(=NC(C)c2nccc(=N)[nH]2)[nH]1 C1(CNC(C2CC(N(C)C)C2)=O)CCC12CN(C(=O)Cc1ccc(F)c(F)c1)C2 c1(CN(CC(=O)NC(CC)CNC(c2cnn[nH]2)=O)C)ccc(CC(N)=O)cc1 N1(C(c2cc(C)ccc2Br)=O)CCN(C(C2C(CC)C2)=O)CC1CO CCCCC(C)C(=O)N1CCN(C2CN(C(c3cc(OC)nc(C)c3)=O)C2)CC1 C1(CNC(C2(OC)CCSC2)=O)CN(C(C2(CC(C)C)COC2)=O)CC(C)(C)C1 c1(C(N(C)CCNC(=O)Nc2cc3sc(Br)cc3s2)=O)cc2ccccc2[nH]1 N1(C(c2c(OC)n[nH]c2)=O)CCNC(C(=O)Nc2cc(C(C)C)n[nH]2)C1 CC1CCN2C1C(=O)NCc1scc(n1)C2=O.C1(NC(=O)N(C)C)COC1 C1(C(=O)NCC2(NC(C3C(C)CC=CC3)=O)CCCCC2)CCCC(=O)N1C N1(C(C2ON=C(C)C2)=O)CC(NC(=O)Cc2ccc3n[nH]cc3c2)CC(C)(C)C1 C1(C(C)C(=O)N(C)Cc2cncnc2)CCN(C(C23CSCC2C3)=O)CC1 C(=O)(CS(C)(=O)=O)NCC1C(C(=O)NC(CC=C)CC)OCC1 C1(C(=O)OC(C)C)CCN(C(=O)NC2CCCC(CO)O2)CC1 c1(C(c2nc(-c3ccco3)nn2Cc2ccc(C)cc2)CC)ccc(F)cc1 C1(NC(C(C)OC(c2ccc(C3CC3)cc2)=O)=O)CCCC(C)(C)CC1 CCCC(C(=O)NC(c1ccccc1O)C)NC(=O)CNc1cccnc1 C(C1Cc2ccccc21)NC(C1C(C)(C)C1(C)C)c1nnnn1C1(C)CC1 CCCCC(O)CCC(=O)N1CC(NC(=O)CCN2C(C)CCCC2C)C1 C1(O)(CCNC(c2nn[nH]c2Cl)=O)CCCN(C(c2cnccn2)=O)C1 C(=O)(C1=C(C)CCCC1(C)C)NCC1CC(NC(C2(OC)CC2)=O)C1 N1(C(=O)NCCCC(C)C)CCCC(C)(C(N2CCC(O)C(C)C2)=O)C1 C1(C2CCOCC2)(CNC(CCCOC)=O)CCN(C(C2CCN(C)C2C)=O)C1 C1(C(=O)Nc2ccc(-c3ccco3)[nH]2)CC(F)CN1C(C1C(C(N)=O)C1)=O c1(CCC(=O)N(C(Cn2cc(C3(O)CCOC3)nn2)C2CC2)C)cccc(F)c1 c1(C2CC(C)(C(N(CC(=O)Nc3ccc(F)cc3F)C)=O)C2)ncc2n1CCCC2 C(=O)(C(O)C(C)(C)CC)NCC1C(CNC(Cn2cc(C(=O)OC)nc2)=O)C1 c1(C(N2C(c3cn(CCC(C)(C)O)nn3)CCC2)=O)ccc(CS(C)(=O)=O)cc1 CC(C)(C)CC(O)CNC(C1(CCNC(=O)CCc2cccnc2)CC1)=O Cn1[nH]nnc1=NCC12CC(CNC(=O)CCCC3CC3)(CO1)C2 c1(C(C)C)cc(C(N2CCN(CC(F)Br)CC2)C(=O)NCCC2CC2)cc(F)c1 N1(CCNC(CCCC#C)=O)CCN(C(=O)CCC(=O)OC(C)(C)C)CC12CCC2 C1(NC(C(C)Cc2cnc[nH]2)=O)CN(C(=O)Cc2cccc(Cl)c2Cl)CCC1C c1(C(CNC(c2c(CCC)occ2)=O)NC(c2cc(C)[nH]n2)=O)cccc(C)c1 N1(C(C2C(C)(CC)C2)=O)CCOC2(C1)CN(C(=O)Cc1ccccc1SC)C2 Cc1cc(F)c(F)cc1C(=O)NCC1CCCN1C(c1ccc(Cl)cc1C)=O O=C(C1=CC2C=CC1C2)NCCC1CC(C(=O)NCC2CC(CC)=NO2)C1 C1(C(C(=O)NCC(=C)Br)NC(=O)C=C2CCC2)CCCC1 C12(NC(c3c(CC)occ3)=O)CC3CCC(C1C2)N3C(c1nocc1C1CC1)=O c1(OCC)cccc(C(N2CC=CC2(C)CO)C(=O)NCCCSC)n1 N1(C(CCCCC(C)C)=O)CCCC12CCCN(C(=O)CC1(CO)CCC1)C2 C1(NC(=O)Nc2c(OCC)cc(C)cc2)CCCC12CN(C(C1CC1(C)C)=O)C2 c1(C(N2C(CCNC(c3cc(Cl)ccn3)=O)CCCC2)=O)occ2c1CCCC2 c1(NCC2(F)CCC2)nccc(N2CCC(C(F)F)C2)n1 C1(CCC(=O)N(c2nccn2C)CC)CN(C(=O)CC(O)Cc2ccccc2)CC1O CC1Oc2ccc(C(N3CC4C(CNC(=O)CC(C)N(C)C)C4C3)=O)cc2C1C c1(C(N(C2CN(C(C(C)C#N)=O)CC23CC3)C)=O)n[nH]c2ccccc12 C1(C(=O)NCC2N(C(CCC(=C)C)=O)CC(O)C2)CCN(S(=O)(=O)NC)CC1 c1(NCC2C(C)(C)C(O)C2)ccc(S(=O)(=O)N2CCC(C)(C)CC2)cc1Cl N1(Cc2cnc(C)o2)CCC2(CCCN(C(C3CCCCCC3)=O)C2)C1 c1(C(N(c2n(CCC)ncc2)C(C)C)=O)nc(C2CCC2)oc1C c1(C(N2CCCCC2CC)C(=O)NCCC)cccc(C)c1F N1(C(C)=O)CCOCC1C(=O)NCC(C)CNC(=O)CCc1cccc(O)c1 C#CC1(NC(=O)CC(C)(C)CNC(=O)CCCC(C)C)CCCCCC1 C1(NC(c2c(Cl)nc(N(C)C)s2)=O)CC2CCC1N2C(=O)CC1CCC(=O)N1C c1(C(=O)NC2CCC(NC(c3cc(C(CC)C)no3)=O)C2)cccc(CF)c1 c1(N(C)Cc2ccoc2)nc(=NCCCC2CC2(Cl)Cl)[nH]c2cc[nH]c12 O=C(CCCCC(F)(F)F)NC(CNC(C1CCC2(CCC2)CO1)=O)CO N1(C(C23CC(NC(C(CSC)O)=O)(C2)C3)=O)CCC(C)=C(C)C1 CC(C)C(CN=c1nc(NCC(C)C#N)c2c([nH]1)CSC2)OCCO C=C=CCCC(=O)N1CCCC1C(C)NC(=O)C(c1ccc(F)cc1)(C)F C1(O)(C(=O)NC2CCCC(NC(=O)CC3(CO)CC3)CC2)CN2CCC1CC2 c1(C(=O)NCCC(C)NC(=O)C(O)CN(C)C)cc(Cl)cs1 Cn1cnc(C(=O)NCC(C)=CC(N2CC(C(C)(C)C#N)C2)=O)c1 N1(C(CC#N)=O)C(CC(N2CCC(O)C2c2ccccc2)=O)C2CCCC12 C1(C(N2CC(CN(C(C(C)Sc3ccccc3)=O)C)C2)=O)CCN(C)C1=O CCCCCCC(=O)NCc1cc(C(=O)NCC2CCC(C)N2C)co1 O=C(N=c1[nH]oc2c1COCC2)NC1CCc2cc(F)ccc2O1 Cc1nccc2c([N+](=O)[O-])ccc(N3CCN(c4nccnn4)CC3)c12 N1(C(C2N(C(C)=O)CCC2)=O)CCOC2CN(C(c3ccnnc3C)=O)CC12 Cc1ccc(F)c(CNC(=O)C(c2cn(C)nn2)NC(C2CC(F)(F)C2)=O)c1 c1(CC)ccc(C(=O)N(C)CCN(C)C(C2(c3ccccc3)CC2)=O)s1 N1(C(C(C)(C)C2CC2)=O)Cc2ccccc2OC2(C1)CN(C(=O)CC1CCC1)C2 CC(C)(CCCC(=O)NCCC1(C)CC1)NC(C1CC(C2CC2)=NO1)=O c1(C(=O)NCC2C=CC(NC(c3cn(C(C)(C)C)nn3)=O)C2)ccc(O)nn1 c1(C(=O)NC2CC(CCNC(c3cc(O)nc(Cl)c3)=O)C2)cncc2sccc12 Cc1nn(C)c(Cl)c1CC(N1CC(NC(=O)CCc2cn(C)nn2)CC1C)=O N1(C(c2c(C(C)C)nns2)=O)CC2CN(C(c3cc(O)c(F)cc3N)=O)CC2C1 O=C(CCS(=O)(=O)c1cccc(Br)c1)N1CCCCC(O)CC1 c1(C(N2C(C)CC(C)N(C(c3csnn3)=O)CC2)=O)ccc2c(O)nncc2c1 C(C(C)(C)CNC(C1C2COCC12)=O)NC(CCNC(C1C(C)C1)=O)=O N1(C(CNC(c2ccc(Cl)s2)=O)=O)CCC(Br)CC1.C12CCCN1C2=O c1(C(c2n(CCCSC)nnn2)NCc2csc(C)n2)cc(C(C)C)ccc1F c1(C(=O)NC2CCC(CNC(=O)CC3OCC(C)(C)C3)C2)cccc2cncn12 C1(CC)C(=O)NCCN1C(C1(CCNC(=O)CCC2CCOC2)CC1)=O CCC(O)C(C)C(=O)N(CC(C)(C)CNC(=O)C(c1nc(F)ccc1Cl)C)CC Cc1cc([N+](=O)[O-])ccc1CNC1CCCC1C(=O)Nc1nccnc1Cl N1(CC(C)C)CCC(C(=O)NC(C)(C)CNC(c2cc(C(F)F)cs2)=O)C1 N1(C(c2ccc(COC)s2)=O)CC2(C1)SCCC2NC(c1csc(C)c1)=O c1(NC(C2CC(C)(NCC(CC)NC(c3ccc(C)s3)=O)C2)=O)cccc(C)c1 N1(C(C(CC)(CC)CO)=O)Cc2ccc(C(C)NC(c3occc3Cl)=O)cc2C1 C(=O)(C(C)(COC1CC1OC)OC)NC(CNC(CCOC)=O)(C)C1CC1 O=C1C(NC(c2nnnn2CC(F)F)c2nccs2)CCN1O N1(C(CCN(CCCCC)C)=O)CCN(C(C2CCC(C)CC2)=O)C2CCC12 Cc1ccc(C(N2CCN(C(=O)Cc3cccc(C)c3)C(C)C2)=O)c(C(C)C)n1 c1(C(=O)NC(C(C)C)CO)nc(NC(c2ccc(OC(F)F)cc2)=O)cn1C CCC#CCCNC(=O)CC(O)C1CCC1ONC(=O)c1ccco1 c1(Oc2c(CN)cccc2)ccc(F)cc1F.c1cc(CN2CCOCC2)on1 N1(C(C(n2cc(C(C)(C)F)nn2)C)=O)CCOCC2(CCC2)C1 CC(CN(C)C(c1cnoc1)=O)N=c1[nH]oc2ccccc12 S(=O)(=O)(c1ccc(NC(CO)CCF)nc1)NC1CC2(CC(OC)C2)C1 C12CCC1CC2.Cc1ncoc1CN(C(C)C(C)(C)C)CCO O=C(C1=CC2CC=CCC12)NCC1=CCN(c2nc(CC3CC3)ns2)CC1 c1(C(C)C(=O)NCCOC2CN(C(=O)C=CC3CC3)C2)ccc(Br)cc1 C(=O)(C1CCCn2ccnc21)NC1(CNC(C2(C)CC(F)(F)C2)=O)CCC1 C1(CCNC(=O)C=CC2CCCC2)CSCCN1C(c1cnn(C(C)C)c1Cl)=O Cc1nc(C(=O)NCc2ccsc2C(=O)NC2(C(N)=O)CC2)sc1C Cn1cncc1C=CC(N1CCCC(CCC(=O)NCC2=CCCC2)C1)=O C(CCC)(CC(=O)N1CCN(C)C(CC)C1)NC(C1N(CCC)CCC1)=O C1(C(=O)NCC(c2ccsc2)C)(CC)CN(C(=O)C(F)CC2CCOC2)C1 C=C1CCN(C(=O)C=CC(C)CC)C(C(=O)N(C2CCCC2C)C)C1 Cc1noc(C)c1CC(C)C(=O)N1CCC1CNC(=O)CCOC1CCOCC1 CCC(O)C(C)(C)C(=O)N1CCC(NC(=O)CC2(C)CCC2)C(C(N)=O)C1 Cc1c(C(=O)NC(CO)C(C)NC(C2CCC3(CCC3)C2)=O)[nH]c2ccccc12 N1(C(CC23C(CN(C(CSC(C)(C)C)=O)C2)CC3)=O)CC2(CCOC(=O)N2)C1 CCC(C)(CNC(C1CC(NC(=O)CCC(C)(C)N(C)C)C(O)C1)=O)C(N)=O N1(C(CCC(=O)OC)=O)CCN(C(c2nc(C)n(C)c2C)=O)C(C)C1C n1(CC)c(CNC(=O)CCC2CCC(NC(c3cnsc3)=O)C2)nnc1O C1(CN(C(COCc2nnc(C)s2)=O)C)CCC(NC(=O)C(C)(C)CO)CC1 N1(C(C(C)CNC(c2cc([N+](=O)[O-])n[nH]2)=O)=O)CCC(C2=NOCC2)C1 C(C(CO)C(C)CC)NC(C1(NC(C2C(=C)C2)=O)CSC1)=O N1(C(c2cc(OC)no2)=O)CCC(C)C1CNC(C1COCCO1)=O C(=O)(C1CCc2ccccc21)NCCC(CC)(CC)NC(c1ccncc1F)=O N1(C(C(C)C)=O)CCOC2C(CNC(=O)CCS(C)(=O)=O)CC12 C1(C)(CC)CC(NC(c2c[nH]c(Br)c2)=O)CN1C(=O)Cc1cc(C)on1 CC1(C)COCCC1C(=O)NC1(CNC(=O)CC2CCSCC2)CCCC1 c1(C(N(C(C)CNC(c2cncc(Cl)c2Cl)=O)C)=O)ccc(O)cc1[N+](=O)[O-] Cc1cc(C#N)ccc1C(=O)N(CCCNC(=O)C(C(C)C)n1cncn1)C c1(C(=O)NCC(C)NC(COCC)=O)cc(C(F)F)cc(F)c1 c1(C(=O)NCCCN(C(c2cc3scc(C)c3[nH]2)=O)C)coc2c1C(=O)NCC2 C1(NC(c2cnc(C)s2)=O)CS(=O)(=O)CC1NC(=O)CC1CCC1 N1(C(CCOC)=O)CCC(CC2CCCN(C(c3cn(C(C)C)cn3)=O)C2)CC1 CS(=O)(=O)C(Cc1ccccc1)C(=O)N1CC2(CC(CNC(C3CC3F)=O)C2)C1 c1(NCC2CCCN(CC(F)(F)F)C2)c(Cl)ccnc1Br Cc1ccc2c(c1)CCC(C(=O)N(C(C)CNC(=O)C=Cc1ccncn1)C)O2 C1(C(=O)NCC=CC(=O)NCCn2cnc(CO)c2)CC2CCC1O2 N1(C(C(CC)=CCCC)=O)CCN(C(=O)C(N2CCOCC2=O)C)CC1CF C1(C2CC2)(CNC(C(=O)N(C)C)=O)CCN(C(c2ccc(Cl)c(F)c2O)=O)C1 C1(CNC(CCCC(C)O)=O)C(C2CC2)CCN1C(=O)CCc1ccncc1 O=[N+]([O-])c1ccc(Cl)c2c1CNC2NC1CCNC(C(F)F)C1 Cc1ccc(Br)c(C(N2CC(CC(=O)Nc3cnc(Cl)c(F)c3)C2)=O)c1 c1(C(N2CCCSCC2)=O)c(F)c(F)c(F)c(F)c1F Cc1ccc(C(=O)NCC2(O)CN(C(c3sccc3Br)=O)C2)c(C)c1Br CC1(C)C2COC1(C(=O)NC1CN(C(c3ccncc3C(F)(F)F)=O)C1)C2 Cc1cc(C(=O)NC2CC(NC(=O)Cc3ccc(O)cc3)CC2O)nn1C(C)C O=S(=O)(c1ccc(NCC)c(Br)c1)N1CCCC(C)C1.C1(C(CF)N)CCOCC1 C1(C(N(C(C)C(=O)NCC2(Cl)CCC2)C)=O)CCCN1CCO N1(C(C2(COC)CCCO2)=O)CCC(NC(C2CCS2(=O)=O)=O)C(C)C1 C(=O)(CCC(CF)CF)N1CC(C)(C)C(NC(c2ccc(SC(F)(F)F)o2)=O)C1 C1(C(=O)N(CCNC(C2(C#N)CC2C)=O)CC2CC2)(NC(=O)OC)CCCC1 c1(OCCOCC(CO)N)ccccc1.CCCCOC(=O)CC c1(N(C(c2cc(CNC(=O)CCc3ccoc3)[nH]n2)=O)CCO)ccccc1 CCC(CC(=O)N1CCN(C(=O)C2=NOC3(CCC3)C2)CC1C)CC(C)C C1(OC)CN(Cc2cc(C(F)(F)F)ccc2C(=O)O)CCC1C C1(C(N2CC(CO)C(C3CC3)C2)=O)CN(C(=O)Cc2cc[nH]c2)CC12CCC2 N1(C(Cc2ccc(C)o2)=O)CCC(C)C(CNC(=O)C=CC(C)(C)C)C1 O=C(C1CCSc2ccccc21)NC1CC(c2nc[nH]n2)N(C(C2COC2)=O)C1 C#CCCCCC(=O)N1CCN(C(c2cc(OC)ns2)=O)C(CO)C1 C#CCC(C)(C(=O)N1CCS(=O)C(C)C1)NC(=O)CCc1cnn[nH]1 C(C)(C(=O)N(CCO)CCNC(=O)C(Cl)Cl)OCC#C C1(F)(CNC(c2c(C(C)(C)C)con2)=O)CCC(NC(C2CCCN2N=O)=O)C1 c1(C(N2CC(CC=C)(NC(=O)C(C)S(C)(=O)=O)C2)=O)cnc2c(c1)CCOC2 C1(CC)(NC(c2cc(C3CC3)nn2C)=O)CCCN(C(=O)CC2CC2)C1 c1(C(N2CC(CC(F)(F)F)C(F)C2)C(=O)NCCCC)cc(OC)cc(CC)c1 c1(N(C)Cc2n(CC)ccn2)nc(N2CC(CC)OC(C)C2)c2c(n1)COC2 c1(C(N(C(CNC(CC(CC)c2ccccc2)=O)C)C)=O)cn2nc(C)sc2n1 C1(NC(CNC=O)=O)CCCCN(C(c2ccncc2N2CCCCC2)=O)C1 CN1CCN(C)C(C(=O)NCC2CCC(NC(=O)CC3CC34CC4)CC2)C1 Cc1nc(C2CCCOC2)sc1CNC(=O)NCC1CC(C(=O)OC(C)(C)C)C1 Cn1cc(CNC(C2CC3CCC2N(C(C2CC2(F)F)=O)C3)=O)c2ccccc12 N1(C(C(c2nc(O)[nH]c(=O)n2)=O)=O)CCn2nc(CNC(C3CCC3)=O)cc2C1 CC(c1ccccc1C)=CC(=O)NC1(CNC(=O)C(O)CC[S+](C)C)CC1 N1(C(c2c(OC)csc2)=O)CC(NC(=O)CN2CCCC(NC)C2)CC12CCC2 c1(C(=O)Nc2scc(-c3cn(CCCC)nc3)n2)ccc(Br)c(Cl)c1 C12(NC(C3CCC4CC4C3)=O)CC3CC(C1)CC(NC(C1COC1)=O)(C3)C2 C1(NC(C(C)N(C(c2cn(CC=C)nc2)=O)C2CC2)=O)C=CCCC1C N1(C(C2C(O)CCN(C(=O)Nc3cccc(C)c3C)C2)=O)Cc2ccccc2C1 N1(c2cc(OC(C)C)ncn2)CCC2(CCCN(C(=O)C(C)(F)F)C2)C1 c1(NC(C)=O)cccc(NC(=O)CCOC(=O)C(C)OC(C)C)c1 c1(C(=O)N(C2(CCNC(CC(C)(C)C)=O)CC2)CCO)cccc(F)c1C(F)F C(C(O)CC(=O)NC1(CC=C)CCCC1)NC(C1(CO)CCCC1)=O C1(NC(c2c(C)nn(C(C)C)c2)=O)CC2CC1N(C(=O)CSC(F)F)C2 C=CC1(C(N2C(C(N3CCC3C3CCCCC3)=O)CC2C)=O)CCCCC1 C(=O)(CCC(CC)CCC)NC(CC#C)(C)C(=O)N(CC(=O)NC(C)(C)C)C c1(CCNC(C2CC2NS(=O)(=O)Cc2cccnc2)=O)ccc(Cl)cc1[N+](=O)[O-] c1(OC)cnc(F)cc1C(N1CCC(CO)(CNC(C2CC23CC3)=O)CC1)=O C1(C(N2CC(F)(CNC(C(C)O)=O)C2)=O)CCCCC1(C)C c1(C(=O)NC(CC)CN(C(=O)CSCc2nnc(C)[nH]2)C)ccc(C#N)cc1O CCS(=O)(=O)c1cccnc1C(=O)NCC1CC(NC(C2C3CCC2CC3)=O)C1 N1(C(COCCOCC)=O)CCN(C(=O)Cc2cc(Cl)cs2)CC2CCCCC12 c1(C(N2C(CN(C)C)CC(O)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C1(C(N(C2CN(C(c3cc(C(C)C)n(C)n3)=O)C2)C)=O)CC(C)OC(C)C1 c1(OC)ccc(F)c(C(N2CCNC(C(=O)NCc3cnccc3OC)C2)=O)c1 Cc1ccc(C=CC(=O)NCC2C(C)CCN2C(C2CC(N(C)C)C2)=O)cc1 N#CC1CCCC1NC(C1CCCN1C(C1CC(=O)CCO1)=O)=O N1(C(C2C(C)C2)=O)CCC(C)(C(=O)N(c2ccc(Cl)cc2)C)C1 c1(C(N2CCC(N(C(=O)C(C)O)CCC)C2)=O)ccn2cc(C(F)(F)F)nc2c1 Cc1n[nH]c(C)c1CCC(=O)NCCN1CCN(C(C2CCCOCC2)=O)CC1 C1(OCC(=O)NC2CCC(CCC(=O)NCc3c[nH]nc3O)C2)CCC(C)CC1 FC1(F)CC(N2CCC(CCCNc3nccs3)CC2)CC1 C1(NC(C(C2CC(F)(F)C2)OCC)=O)(COC)CN(C(C2CC2C)=O)C1 C#Cc1ccc(C(=O)NCCCN(C(c2nocc2Br)=O)CC)c(OC)c1 CCCC(O)C(=O)N1CC=CC1CNC(=O)CCCc1ccccn1 C#Cc1cc(C(=O)NCC2CC2CNC(c2[nH]c(C3CC3)nc2C)=O)cc(N)c1 c1(C(=O)NC(CC(C)NC(Cn2c(C)c(Cl)cn2)=O)C)n[nH]c2c1COC2 c1(CC(C)NC(=O)CSc2ccc(F)c(F)c2)cccc2c1OCO2 CC1CN(C(=O)C(=O)Nc2cnns2)CCC1C(=O)Cc1ocnc1C(F)(F)F C1(NC(C(CC=C)OC)=O)CCN(C(c2coc(C(F)F)c2)=O)C12CC2 C1(O)(CNC(c2cc(CC)no2)=O)CCCN(C(=O)C(C)NC(C)(C)C)C1 c1(C(=O)OC(C)(C)C)ccc(NC2CC(CN)C2(C)C)c(N)c1 c1(C(=O)NCCOCCN(C(C2CC(C)OC2)=O)C)nc(Cl)c(Cl)s1 c1(C(N2CC3CC(NC(=O)C4=CCCOC4)CC3C2)=O)cncc2cnccc12 Cc1cn(C(C)(C)C(=O)NC2CC(NC(=O)CC3CC3(Cl)Cl)C2)cn1 c1(C(=O)NC2CC(C)N(C(c3ncn4c3CCC4)=O)C2)c(Cl)cc(Cl)nc1N C1(CC(=O)N(CC(COC)C)C)CC(C)(C)CN1C(=O)COCC1CCOCC1 CC#CC1CCN(C(C2(C)C=CCN2C(c2ccncc2CC)=O)=O)C1 c1(OCC)c(C(=O)NCC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)cccc1F C12(COC)CC(NC(c3cccn3C(C)C)=O)(CN1C(C1CC1C)=O)C2 C1(C(N(CC(NOC(COC)COC)=O)C(C)C)=O)CCCC1C1CC1 CCCCC(C)C(=O)NCc1n[nH]cc1C(=O)NCCC1CCCN1C c1(C(=O)NCC23CCN(C(C(C)=O)=O)C2CCC3)cc(C)nc2ncnn12 C1(NC(=O)NC(CCC)COC(C)(C)C)CN(C(=O)OCC)CCS(=O)(=O)C1 c1(C(=O)NCCOCCOC)oc(CNC(c2cnc(C)n2C)=O)nc1C Cc1c(C(=O)NC(C(N2CCC(F)(C#N)C2)=O)c2ccco2)cncc1F c1(CC(N2CCC(NC(=O)CC3OCCCO3)(CF)C2)=O)ccc(Br)cc1F c1(C(=O)OC)cncc(CNC(=O)N(C)CCC2CCC2)c1 CC1C(NC(C2CCCC2)=O)CCCN1C(=O)Cn1cc(CO)nn1 C1(C(N(CC(COC)O)C)=O)CCC2(CC2)N1C(=O)CC(C1CC1)C1CC1 CCC(O)C(C)(C)C(=O)N1CC(CNC(C2(CF)CCOCC2)=O)C(F)(CO)C1 CC1CN(C(C2(O)COC2)=O)CC1(C)CNC(C1CC2C=CC1O2)=O C(CCC(C)C(=O)NC(C)CCCNC(=O)Cc1cncn1C1CC1)OC N1(C(Cc2cc(C)on2)=O)CCCC(C2CCCCN2C(=O)CN(C)C(N)=O)C1 c1(OC)ccc(OC(F)(F)F)c(CNC(C2CC2NC(C2CC=CC2)=O)=O)c1 N1(C(CC2(OC)CCCC2)=O)CC(NC(=O)CSc2n[nH]c(O)n2)C(F)C1 c1(CCNC(NC(C(=O)OC)(C)C)=S)c[nH]c2cc(Cl)cc(Cl)c12 CC1CCC=C1C(=O)N1CCC2(CC2NC(C2C=CCS2)=O)C1 C1(CNC(C(C)(C)CF)=O)CC2(CCN(C(=O)CC3CCCCC3)C2)CO1 c1(C(=O)NC(C2C(C(N(C3CCC3)CC#C)=O)C2)C)cc(C2CC2)on1 c1(C(N2C(CC(=O)Nc3ccnn3CO)CC2)=O)nccnc1-c1ccccc1 N1(C(C2CCC(SCC)CC2)=O)CC2CC1CN(C(=O)Cc1cscn1)C2 C(=O)(CCCC(C)(C)NC(=O)CC1CCCOC1)NCc1ccc(C)cc1F C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C(Cc2ccc(S(C)=O)cc2)=O)CC1 C(=O)(CC(C)CC(=O)NC1CCC(CCNC(=O)C2=CCOC2)C1)OC C#CC1(C(=O)NCCS(C)(=O)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C1 Cc1nn2c(c1C(N1C3CCC1CN(C(C14CCCC1CC4)=O)C3)=O)CCCC2 C(C1CCc2ncnn21)NC1C(C)CCCCC1 C1(NC(C(c2ccccc2)C)=O)COCCN(C(c2c(C3CC3)noc2C)=O)C1 c1(C(N2C3C(NC(C(CC)NC(N)=O)=O)C(CC3)C2)=O)cnc2cc[nH]c2c1 N1(C(C(=O)NC2CC2)=O)CCCCC1CCNC(C1(F)CCCOC1)=O N1(C(C2C(C=C)C2)=O)CCC2(C1)CN(C(=O)C(C1CC1)SC)C2 Cc1nc(CCC(=O)NCc2nc(CO)n(C)n2)[nH]c1C CC(CC(N)=O)C(=O)NC1CC(NC(c2cnc(C(C)C)[nH]2)=O)C1 C1(CNC(c2c(C)nc(O)[nH]2)=O)CN(C(=O)Cn2c(C)c(C)sc2=O)CCN1C c1(C(N(CC(CNC(C(C)OC2CCCC2)=O)O)C)=O)cnc(S)[nH]1 c1(C(=O)NCCC(C)NC(c2nc[nH]c2C(C)(C)C)=O)ccc(N)cc1 C(=O)(C(O)C1=CCCCC1)NC1CC(CC(N2CCC(C)CC2)=O)C1 C12(CNC(Cc3n(C)ncc3)=O)CC1CN(C(=O)Cc1csc(Br)c1)C2 c1(C(=O)NC2CCN(C(c3c(CC)con3)=O)CC2C)nncc2c1CCCC2 c1(C(=O)NC(CC)(C)CNC(=O)C(O)CCSC)cc(OC(C)C)ncc1Cl CC(=O)CCCC(=O)N1CCCC1C=CC(N1CCOC(C)(C)C1)=O c1(NC(=O)Nc2cn(CC)nc2)cccc(Cl)n1 C1(=O)CCCCN(C)N1CCOCCCC(F)(F)F.CS Cc1nn(C)c(C)c1CC(=O)NCCCCNC(=O)CC1CCC(O)C1 c1(CC)ccc(O)c(C(N2CCC(NC(c3ocnc3C(F)F)=O)C(F)C2)=O)c1 N1(C(C2(C)CCCN(C(C3CCCC3)=O)C2)=O)CCCC2CCCCC12 C(=O)(C=C1SCC(=O)N1C)NCC1N(C(c2nc(CC)oc2)=O)CCC1C1CC1 CCC(CNC(=O)CC1CCC(=O)N1)(CC)C(=O)N1CCC1CN=[N+]=[N-] C1(C(=O)N(C)Cc2cn(C)cn2)(CNC(C2CN(C(C)C)C2)=O)CC=CC1 CC1(C(=O)NC2(CNC(C3CC(CC4CC4)C3)=O)CCC2)CCOC1 N1(CC(=O)NC2(C)CC(NC(c3cn(CC=C)nn3)=O)C2)C(=O)CC(C)(C)C1=O CC(C(C)(C)C(=O)N(C)CCC1CC1)NC(C1C2CCCCC12)=O CC1CCC(=CC(N2CCC(NC(=O)C(c3ccc(Cl)nc3)(F)F)C2C)=O)CC1 c1(N2C(C3CCN(C(C4CC(C)(F)C4)=O)C3)CCC2)ncc([N+](=O)[O-])cc1Cl C1(NC(C2N(C(CCC)=O)CSC2)=O)CN(C(=O)CCC2CCCN2C)CC1C CC1CN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)CC(C)(C)O1 C12(CNC(C#CC(C)C)=O)CN(C(=O)CN3CCC(C)(O)C3)CC1CCO2 C1(C(=O)NCCN(CCOC)C)CC2CCN(C(=O)C(C)(O)C(C)C)CC12 N1(C(=O)NCCC(F)CO)CCOC(C2CC(F)(F)C2)C1 c1(CCC)ccc(C(=O)N(C2C3CN(C(C4CCCN4C)=O)CC23)C)cc1 C1(O)(C(N2CC(CN(C(=O)COC(C)(C)C)C)C2)=O)CCOCC1 N1(C(CC(CC)CN(C)C)=O)CCCC2(NC(C3(C4CCCO4)CC3)=O)CC2C1 c1(C(N(CC(O)CN(C(=O)C(F)OC(F)(F)F)C)C)=O)cnccc1C(F)F CC(CCCCNC(=O)C(C)n1cccc1)NC(=O)Cn1cnnc1O CC(C1CCCCC1)=CC(=O)NC(c1ccccc1)CNC(c1[nH]ccc1C)=O C1(NC(c2cnc(CC)s2)=O)CCCC(NC(c2cn(C3CCC3)nc2C)=O)C1 C=CCCCC(C(=O)NC(C1CCCC1)(C)C)NC(=O)CC1CCOC1 N1(C(C(CC)CC)=O)CCC2(C)CN(C(C3CC3Cl)=O)CC12 C1(C(C)C)CN(C(=O)C=C2CCN(C)C2)CCN1C(c1ccc(F)c(CO)c1)=O C(=O)(C(O)(C(C)C)C(F)(F)F)NCC1(NC(C=COCC)=O)CCCCC1C C(=O)(C(F)(F)Cc1cn(CCCN(C(=O)C(F)OC(F)(F)F)C)nn1)OCC c1(C(=O)NCC2C(NC(c3occc3Br)=O)CC2)cccc2ccnn12 C1(CNC(C2CCC=CCC2)=O)CC12CCN(C(C1CC3(CCCC3)C1)=O)CC2 Cc1cccc(CC(=O)NC2CC3CCC2(NC(c2ncn(C)n2)=O)C3)c1Cl CCCC(CNC(C1(OC)CCN(C(c2cc(C)nn2CC)=O)C1)=O)CCC Nc1cc(Cl)ccc1C(=O)NCCCCNC(=O)CCCC1CCOCC1 C1(CN(C(=O)C(C)N2CCCC2)CC)CCN(C(C2C=CCCC2)=O)CC1 C1(C(N2CCC(C(=O)NC)C2)=O)(COC)CCN(C(c2cncc(C)n2)=O)C1 C(=O)(C1CCCc2ccnn21)N1C(CNC(C(C)(C2(C)CC2)NC(C)=O)=O)CC1 CC1C2CCCCC2CN1C(=O)C(c1ccnn1C)NC(C12CC1CNC2=O)=O C1(NC(CC(C)c2ccccc2)=O)CN(c2nccc(CO)n2)CC1F Cc1ccc(C=CC(N2CC(C(O)C(N3CCC(N(C)C)CC3)=O)C2)=O)o1 N(C1=NCC2(CCC2)CN1)C(COC)C.C1(SC(C)(C)C)CCOC1 N1(C(CCC=CCC=C)=O)CCN(C(=O)Cc2ccnn2C)CC1CC(=O)NC C(=O)(CC(C)CC(F)(F)F)NC12CCN(C(CCCC(=O)OCC)=O)C1CCC2 N1(C(COC(CC)C)=O)CCCC1CCCNC(c1n[nH]cc1C(F)(F)F)=O c1(NC(C)=O)cscc1-c1c[nH]c(C(=O)N(CCN(CCSC)CC)C2CC2)c1 c1(C(C)(CC2CCCC2)OCC(=C)Br)nnnn1CCCC C1(N(C(C(CC)(F)F)=O)C)CCCN(C(=O)CC2CCC(=O)O2)CC1 C(=O)(C(F)C(F)(F)F)NC(C(=O)NCc1cnn(CCF)c1)Cn1cncn1 C=C1CCN(C(c2ccc[nH]2)=O)C(C(=O)NCC(C)N=[N+]=[N-])C1 C1(C(N2C(CC(=O)NCc3csc(Cl)n3)CC2)=O)(CO)CCCCCC1 CC1C(NC(=O)Cc2ncsc2Cl)CCN1C(=O)CC1CC=CC1 C1(C)(NC(CC2(OC)CC2)=O)CC(NC(C2CCC(O)C2)=O)C1 C1(N=c2[nH]nc(-c3ccccc3)o2)(CC)CCN(C(=O)C=CC=CC2CC2)CC1 Cc1ccc(=O)n(CC(=O)N(C)CC2CN(C(c3cnns3)=O)CC23CC3)n1 CCCC(CCC)C(=O)N1CCCC(c2ccc(CNC)cc2)C1 c1(NC(C2C(NC(c3cc(I)c(F)cc3F)=O)C2)=O)c(F)c(F)nc(F)c1F c1(C(=O)NCCN(C(=O)C(C2CC2)OC)CC)cc(Cl)cc(Br)c1N n1(CC)nc(C)cc1C(N1CC(CNC(=O)C(C)NS(=O)(=O)CC)C(C)C1)=O C1(C(=O)NCC(CC)C#N)CN(C(=O)CN2CCN(C)CC2)C2(CCC2)C1 C1(NC(c2ccc(C)c(CO)c2)=O)CCN(C(C2CCC2(C)C)=O)CC(C)(C)C1 C12(NC(=O)C=CCF)CC3CC(C1)CC(CNC(=O)CNc1nccs1)(C3)C2 N#CC1CCC(CC(=O)NC2(CCNC(=O)Cc3ccccc3Cl)CCC2)C1 c1(C2C(C(=O)NCC3NCC(C)(C)C3)C2)cc(Br)ccc1F C1(CNC(COC(CC)C)=O)CCCN(C(=O)C2=C(Cl)CC2)CC1 C1(CNC(C(CC=CC)NC(c2ccc(CN(C)C)o2)=O)=O)CCC(=O)NC1C N1(C(CCCOC(C)=O)=O)CC(CNC(C2CC(C)(O)C2)=O)C(C)(C)C1 C1(C(N(C2CCN(C(c3n(COC)ncc3)=O)C2)C)=O)CC(F)(F)CCC1(C)C C1(CC=C)(C(=O)NC(CNC(=O)C(F)=CC2CC2)CC=C)CCOC1 c1(NC(C2(NC(C(CCC)F)=O)CCSC2)=O)ccc(C)c(F)c1 c1(C(N2CCC(CNC(C(F)OC)=O)C2)=O)cc(C#N)c(C)cn1 c1(C(=O)NC2C(NC(c3c(C(C)(C)C)noc3)=O)C2)ccnc2ccc(F)nc12 C1(F)(C(N(CCC(=O)NCCn2c(CC)nnc2)C(C)C)=O)CCOC1C c1(C(=O)NC(C2CC(NC(CC3(NC(C)=O)CC3)=O)C2)C)cc2ncccc2s1 c1(C(=O)NCCC2CC(NC(C3CCC(F)C3)=O)C2)nccc2occc12 c1(OC)ncnc(NC(C2CC3CC3N2c2nnc(C(C)C)o2)=O)c1OC N1(C(CC(C)OC)=O)CC(C)(C)CCC1CNC(=O)CC1CCC(C)(O)CC1 O=C(N1OC2CCC1CC2)C1Cc2ccccc2S1(=O)=O c1(OC)cccc(-c2cn(CC(CNC(c3cccnn3)=O)OC)nn2)c1 c1(OC)cc(C(=O)NCC(N2CC(C)OC(C)C2)C(C)C)sc1S(N)(=O)=O C1(C#CC(=O)N2CCCC(C)(CNC(=O)C(O)C(C)(C)C)C2)(CC)CC1 Cc1ccc(C(N2CCN(C(=O)CSC(C)(C)C)CC2CF)=O)c(N)c1C Cc1cc(C(=O)N(CC(C)NC(=O)CSCC(C)C)C)sc1-c1ccccc1 O=C(N=c1ccnc(N2CCCC(CO)CC2)[nH]1)N1CCC(c2ccccc2)C1 Cc1cccc(=O)n1CC(C)(O)C(=O)NCCCCC(C)NC(=O)C1=NOCC1 CCCCC(C)(F)C(=O)NC(C1CCCCC1)C(=O)NCCCC(=O)NO c1(CN2CC(C(=O)Nc3cnccc3Br)OCC2)cc2ccccc2[nH]1 c1(OC)cc(F)c(F)cc1NC(=O)NCc1cc(F)c(F)cc1O c1(NC2(CNC(C(C)OC)=O)CCCC2)ncc(-c2cnsc2)cn1 c1(NC(C(CCSC)NC(CCCC)=O)=O)cc(C)c(F)c(C)c1 C=Cc1cnn(C)c1C(=O)NC1COCCC1NC(C1CN(C(N)=O)C1)=O C(=O)(CC(O)CCC(C)CC)N1CC(NC(C(C)SCCCC)=O)CC(C)(C)C1 C(=O)(C#CC1CCOCC1)N1CC2(CNC(CCC(=O)N(C)C)=O)C(C1)CCO2 N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)Cc2nc(C(F)(F)F)n[nH]2)C2CCC12 CCCC(C(=O)NCC(C)OC(F)F)NC(C1CCCN1CCC)=O C(c1cncc(O)c1)=C1CCN(C(=O)NC(Cc2ccccc2)CO)CC1 c1(C(N2CC(C(N)=O)(CNC(c3nc(CC)sc3)=O)C2)=O)nc(=O)n(C)[nH]1 C(CC)(C(=O)NC(C)CCCNC(C1CC(C(=O)OC)C1)=O)OCC c1(OC)ccc(Cl)cc1N1CCN(C(=O)NC(C)CCC2CCCCC2)CC1 N1(C(CCCC=C)=O)CCC(O)C(NC(c2cc(Cl)cnc2OC)=O)C1 N1(C(C(n2cc(Cl)cn2)C)=O)CC=C(CCNC(c2nocc2C2CC2)=O)CC1 c1(C(N(CC(C)O)CCNC(C(C)OCC)=O)=O)cccc(C)c1O C1(C)(N(S(C)(=O)=O)CCN(C)C(c2ccncc2)=O)CCCN(CCO)C1 c1(OC)c(C(N2CCCC(CN(C(=O)Cn3cncc3C)C)C2)=O)csc1C c1(C(=O)NCC(C)N(C)C(c2nc[nH]c2C(C)(C)C)=O)ccc2c(c1)CCO2 CCC(C#N)C(=O)N1CCN(C(=O)C(n2ccc(C3CC3)n2)C)CC1 C12(C(=O)NC3CC(F)C3)CCCC1CN(C(C1C=CCS1)=O)C2 c1(C(=O)NCCCCC(C)NC(C2(c3c(C)cno3)CC2)=O)ccccc1S(C)=O n1(CCC(N2CCC(NC(=O)CC3(C(F)F)CC3)C2)=O)cc[nH]c(=O)c1=O c1ccn2ncc(CNc3nc(C4CCCCC4)cs3)c2c1 Cc1cnc(C2CC2NC(C2(O)CN(S(C)(=O)=O)C2)=O)s1 C1(C(=O)NC2C(NC(c3n(CC#C)ccc3)=O)CC2)CCC2CC1C2(C)C c1(C(N2CCN(CCN(C(C(COC)(C)O)=O)C)CC2)=O)cc(F)ccc1C Cc1c(C(N2CCC(C)C(N(C(=O)C=Cc3cccnc3)C)C2)=O)nn(C)c1N Cc1cccc(C(C)C(N2CCC(O)(CNC(c3ncccc3F)=O)C2)=O)c1 C(C)(C)(CC(C)N=c1cccc(S(=O)(=O)N2CCCCC3(CCC3)C2)[nH]1)OC c1(C(=O)NC(COCC)C(=O)NCCC2(N(C)C)CCC2)cnc(O)cc1C c1(C(=O)NCCNS(c2c(C)cc(F)cc2)(=O)=O)ccc2c(C)c[nH]c2c1 c1(OCC(N2CC(CNC(C(C)OC)=O)OCCC2)=O)ccc([N+](=O)[O-])cc1 CCC(C)(C(=O)N(CCCNC(C1COC(=O)C1)=O)C)C(N)=O c1(C(=O)NCC(C)(C)CNC(=O)CCC(=O)N(C)C)cccc(P(C)(C)=O)n1 Cc1cc(F)ccc1C(=O)NCC1CCCN(C(C2CCCCS2(=O)=O)=O)CC1 C1(NC(C2N(C(C)C)CCC2)=O)CC2(C1)CC2NC(=O)CCSc1ccncc1 c1(C(N2CCN(C(CC(C)C(F)F)=O)CC2)=O)coc(C#Cc2ccccc2)c1 c1(C(=O)NCC(N2CCN(CC)C(=O)C2)=O)ccc2c(c1)CCC(O)C2 C12(NC(C3C(C)(C)C3)=O)CCCC1CN(C(C1CCCN(CP(C)(C)=O)C1)=O)C2 CC(C)CCCC(=O)N1CCCCC1(C)c1ccccc1 C1(NC(C(C2(C)CC2)NC(C(CC=CCC)C)=O)=O)CC2C=CCC(C1)C2 N1(C(CC(=C)Br)=O)CC(C)C(NC(=O)CN2C(=O)NC(C)(C)C2=O)C(C)C1 C(C(C)(C)C(=O)NCC(F)(F)Cn1cc(C(=O)NC2CCN(C)CC2)nn1)OC c1(NC(N)=O)cc(Cl)c2[nH]c(-c3cccnc3)nc2c1 N1(CC(=O)OC)CC2(CCC(CNC(c3ccc(CSc4nccs4)o3)=O)O2)C1 c1(C(=O)NCC(n2cc(CCC3CCCC3)nn2)C)ccc(Br)cc1Cl C(C(N=c1cnc(F)c[nH]1)C1CC1)NC(C(C)OC1CCCC1)=O n1(CC)nc(C)c(CNC2(c3nnnn3C(C)(C)C)CCC2C2CC2)c1C c1(C(=O)NC2C(NC(C(C)(C)C#N)=O)CC2)nnn2c1CCCC2 C=CCC(CNC(=O)CNC=O)NC(=O)CC1CS(=O)(=O)C1 c1(C(N2CCC(CNC(C(C)SC)=O)CC2C)=O)ccc2cc(O)ccc2c1 N1(C(CCC(=C)C)=O)CC2CCC2(NC(=O)Cc2cnccc2C)C1 N1(C(C2(C)CC2(F)Cl)=O)CC2CC(C1)C2NC(=O)CC1CC1 C(=O)(CCCOC)N(C(C)CNC(c1cc(-c2ccco2)c[nH]1)=O)CC C1(C(=O)NCCC(CNC(=O)CCSC)NC(N)=O)(CC)CCNC1=O C1(C2(O)CCC2)(C(=O)NC2CC(NC(C=Cc3n(CC)ncc3)=O)C2)CC1 N1(C(C23CCC(NC(CCOCCOC)=O)C2C3)=O)CCCN(CCO)CC1 c1(OC(C)C)nc(N2CCC(NCc3cnc(O)c(Cl)c3)C(O)C2)ncc1Br CC(CC(F)(F)F)C(=O)NC1CC(C)(NC(=O)COc2ccccc2F)C1 N1(C(=O)NCc2c(C)ocn2)CCC12CCCCC2 c1(C(N2CCC(C(=O)NCCOCc3ccccc3)CC2)=O)cccc(I)n1 Cc1ccc2oc(C(N3CC4CCC4(NC(c4ccc(Cl)cn4)=O)C3)=O)cc2n1 C12(COC)CCC(C(=O)NCC3CCC(NC(=O)Cn4cccn4)C3)(CO1)C2 C(=O)(C#CC(C)(C)CNC(C1CCSC1)=O)N1CC(N(C)C)C1 C1(C(=O)NCCOCC(F)(F)F)CC12CCN(C(=O)CCc1ccco1)C2 c1(-c2cnc(N)nc2)c[nH]c2nccc-2c1.Oc1ccc(CN2CCOCC2)cn1 N1(C(=O)NCCCCOCC)CCC2(CC1)CN(C)C(=O)O2 N1(C(c2cccc(C#C)c2F)C(=O)NCC(=O)OC)CCc2ccc(O)cc2C1 N1(C(C(C2CCC2)OCC)=O)CC2CCC2(C(=O)NCC2(C)CC(C)(C)C2)C1 Cc1ncsc1CC(=O)N(C)CC1CCCC1NC(=O)C(O)C1CCC1 CC(C)(C)CC(C)(C)C(=O)NCC1(NC(=O)Cc2ccccc2Br)CC1 C(=O)(C(CC#CC)NC(=O)CC(C)CN(C)C)NCCSCC#C c1(CC(N2CC(NC(CN(C3CC3)CC)=O)C(O)C2)=O)cc(Cl)ccc1OC c1(C(N(C2CCC(NC(=O)CCC3CC3(F)F)C2)C)=O)cc(C(N)=O)no1 c1(NC(C2CCN(Cc3cccc(C(F)(F)F)n3)C2)=O)cc(F)c(F)c(F)c1F CC1(C)CC2(CC2C(=O)NCC2(CNc3ncnc4scnc34)CCC2)C1 Cn1nnc(C(N2CCC(C(F)CNC(C3CC3(Cl)Cl)=O)CC2)=O)c1C(F)(F)F C1(CNC(=O)NCC(=O)Nc2ccc(CCF)cc2)CCC2(CC2)CO1 Cc1cn2cc(C(=O)NC3CN(C(=O)CCn4ccnc4)CC3C)cc(F)c2n1 C12(C(=O)NC3C=CCN(C(C=Cc4c(C)n[nH]c4)=O)C3)CCC(CO)(CC1)CC2 C1(NC(C(C)(C)C2(O)CCC2)=O)CCOCC1C(=O)NCC(N1CC=CC1)=O C1(NC(C2(C)CCC2)=O)CC(O)CN(C(c2cncn2-c2ccccc2Cl)=O)C1 C1(CCC(=O)NCCC(C(=O)OC)C)CCCCN(C(c2c[nH]c(C#N)c2)=O)C1 CCCC(C)(C)CC(=O)NCC1C(C)CCN1C(c1ncccn1)=O N1(C(C2(C(=O)OCC)CC2)=O)CCC2(NC(=O)NC)CC2C1.N12CCC1(C)C2=O O=C(CC1NC(=O)c2ccccc21)NC1CC(CNC(=O)C2=NOCC2)C1 c12cccc(F)c1C(=O)N2.Cc1ncc(CN2CCC(OC(F)(F)F)CC2)cn1 c1(CNC(N2CCC(OCCOC)C(O)CC2)=O)cccc2c1nnn2C C(CS(=O)(=O)C1CCCC1)N1C2(c3n(C)ccc3)CC(CC1)C2.c12nc(n[nH]1)C2OC N#Cc1c[nH]c(=NC2CCC(C(N3CC4CC4C3)=O)OC2)c2ccsc12 N1(C(c2c(Cl)cc(C)s2)=O)CCC(F)(CNC(=O)CSC2CC2)CC1 O=C(CCC(=O)c1ccccn1)Nc1nnc(S)s1.c1(C2CCOC2)ccc(Br)cc1 c1(CNC(C(CC)C)=O)cccc(NC(=O)C(C)CN2CCCCC2)c1 C1(NC(C(C(CC)C)C)=O)CC2(CCN(c3nc(Cl)ncc3C(N)=O)C2)CO1 c1(OC)cc(C(N2CC3CC2CN3S(=O)(=O)CC2CCC2)=O)cnc1Cl C1(NC(C2CCOCC2)=O)CC2CN(C(c3ccnc(Cl)c3F)=O)CC12 CS(=O)c1nc2ccc(C(=O)NNC(=O)Cc3ccc(O)cc3)cc2[nH]1 C(C(CC(F)(F)F)NC(C1CCCS1)=O)NC(CCNC(=O)CO)=O c1(CNC(c2ccc(OC)s2)=O)ccc2c(c1)CN(C(=O)CN1CCC1C)C2 c1(C(=O)NC2CCC(N(C(C(CCCC)C)=O)C)CC2)cnn2ccnc(N)c12 CC1CCN(CC(=O)NC2CCC(CC(=O)N(C)CC3CC3(F)F)C2)C1 C(CN=c1cc(-c2ccccc2)n(C)[nH]1)NC(C(c1cccc(OC)c1)C)=O c1(C(NOCC(=O)OCC)=O)conc1C(C)NC(=O)CC1CCCO1 CC1CN(C(=O)COC2CC2(F)F)CC1NC(=O)CCc1cncc(C(N)=O)c1 c1(OC)cc(C(=O)NCC2CC(C)(C)CN2C(=O)C=C2CCCCC2)ccc1Cl C1(C(N2CC(N(C(=O)C=CCO)C)C2)=O)CC12CCCOC2 C1(CNC(C(C)c2cccs2)=O)CC2CCC(C1)N2C(=O)C(F)C(C)(C)O C1(OC)CCC2(CCN(C(=O)CC3C=CC(NC(=O)CCC(C)(C)C)C3)C2)C1 c1(C(=O)NC2CCN(C3CC3NC(COCCOCC)=O)C2)ccc(F)cc1.C(=O)N.C.CC c1(OC)cccc(C(=O)N(CC(C)NC(C2CC23CCCC3)=O)C)c1 c1(OC)ccc(C(C(F)(F)F)NCCC(=O)Nc2cccc(Br)c2)cc1F C(=O)(C#CC1CCOC1)NC1CC2(C(C(N3CC(O)(CC(C)C)C3)=O)C2)C1 C(N=c1nc(C)nc2[nH][nH]cc1-2)C1(OC)CN(C(c2nnn(C(C)C)c2C)=O)C1 c1(C(N2CCC(C(=O)NC(c3cn(C)nc3C)C)(CC)C2)=O)nccc(C)c1N N1(C(CN(C(C(CC(=O)OC)C)=O)CC2CC2)=O)CCN2CC(C)CC2C1 Cc1cc(C(N2CC(F)(F)CC2(C)CO)=O)c2c(C)nn(C)c2n1 N1(C(C2CCC(C)O2)=O)C2CCC1(CNC(=O)CC1(CO)CCOCC1)CC2 N1(C(CCC#C)=O)CCN(C(CNC(=O)C(N2C(=O)CCC2=O)C)C(F)F)CC1 C1(C(=O)NCCc2n(C)ncn2)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CCO1 N1(C(CCc2c(C)noc2C)=O)CC(NC(c2cccnc2O)=O)CC2(CC2)C1 N1(C(C2(CC)CCCC2)=O)CCCN(C(=O)C(C)COC)C(c2ccccc2)C1 c1(C(=O)NC(C)CNC(=O)C(C)OCc2ccccn2)ccc(C(F)F)s1 Cc1ccc2c(c1)CN(C(=O)C1=NOC(CNC(C3CCS(=O)(=O)C3)=O)C1)C2 N1(Cc2ccc(C(=O)OC)o2)CCN(C(C2CC(CSC)C2)=O)C(CC(C)=O)C1 c1(N(C)CC2(O)CN(C(=O)NC(C3(C)CCC3)C)C2)ccccn1 c1(C2(C(N(CCCNC(C3CCC3C)=O)CC)=O)CC2)ccccc1Cl CCCC(CC)CCC(=O)N1CC2C(NC(=O)CC3=CCN(C)CC3)C2C1 CCC(C)CC(C(=O)NCCOC(C)C)NC(=O)Cc1ccco1 CC(C)C(O)CNC(=O)C=CCN(C)C(C1CC=CCC1)=O N1(CCC(=O)Nc2c(OCC)cccc2)CCCC(NC=O)CC1 Cc1cnccc1CC(C)NC(=O)NCc1nnc(C2CC2)n1C1CC1 C1(C)(OCC)CCCN(C(C23CC4CC2C3C4)=O)C1.C1(C)C(=O)N1 c1(CN(C(=O)NC(=O)C(C)(C)F)CC)cnn(CCc2ccccc2)c1 N1(C(C2(CC(=O)OC)CC2)=O)CC2CCC(CNC(C3CC(C)(C)CO3)=O)(C2)C1 C1(CN(C(=O)CC2OCCO2)C)CN(C(=O)C(N2CCCC2)C2CC2)CCO1 C(CCCCNC(c1cc(C(F)(F)F)on1)=O)NC(=O)C=CC=C(Cl)Cl C12(CNC(C=C(CCC)C)=O)CCC(NC(=O)C(O)CSC)(CO1)C2 c1(C(=O)NCCN(C(C2C(OC)CC2)=O)C)c(Cl)ccc(Cl)c1O C1(C(=O)OC(C)C(=O)NC2CCCC2)CCC(c2ccccc2)C1 C1(NC(C2CC(C)N2C(C2CN3CCC2C3)=O)=O)(CF)CCOCC1 c1(-n2cc(C3CCN(C(=O)CC4CC=CCC4)CC3)nn2)cccc(Br)c1 N1(CC(C)O)CCC(NC(c2cc3n(n2)CCC3)=O)C(O)C1 N1(C(c2n(CC)ccn2)=O)CCC(O)(C(C)NC(=O)C=CI)CC1 N1(C(CC2(OCC)CCC2)=O)CCCOC(CNC(=O)Cc2ccon2)C1 C#CCCCCCC(=O)N(C1CC(C(=O)N(CC(C)CCC)C)C1)C c1(NC(=O)NC(c2ccc3c(c2)CCC(=O)N3)C)c(I)cc(Br)c2ccccc12 c1(C(N2CC3C(C(=O)NCCC4CC(C)C4)(C3)C2)=O)ccc(O)c([N+](=O)[O-])c1 Cc1nn(C)cc1CC(=O)NCC(CC(C)C)NC(c1cnn(C)c1Cl)=O c1(CC)cccc(C(N2CCC(C(N3CCC3(C)C)=O)C2C)=O)c1 N1(c2ncc(C)s2)CC2C(C(=O)Nc3cccc(C(F)F)c3)C2C1 CC(CCC(F)F)OC(=O)Cc1ccc(-c2ccccc2Br)cc1 Cc1nccc(C(=O)NC2CCC(CCNC(c3c(C)noc3N)=O)C2)c1C C1(CNC(C#CC(C)C)=O)COCCN(C(c2cc(Br)sc2Cl)=O)C1 N1(C(CC(=O)OCC)=O)CCC(O)C(NC(c2cncc(SC)c2)=O)C1 C(=O)(C(C(C)C)n1cc(Br)cn1)NCC(C)NC(COCCCC#C)=O C1(CCC)CCC(C(=O)NC2CCC(C(=O)N(C)C)CC2)CC1 N1(C(CC2C(C)(C)C2(C)C)=O)CC2CCC1C(NC(c1cc(C(N)=O)[nH]n1)=O)C2 N1(C(CCCC)=O)CC2CCC1C1CN(C(=O)Cn3cc(C(F)(F)F)cn3)CC21 C=CCCC(F)(F)C(=O)N1CCC(F)(CNC(c2cncc(F)c2Cl)=O)CC1 N1(C(=O)OC(C)(C)C)C(C(N2CCCC2CNC(=O)CC2CCCC2)=O)C1(C)C C1(NC(CC(C)c2ccco2)=O)CC2CN(C(c3ccc(O)nn3)=O)CC2C1 C(=O)(C1=CC2(CCOCC2)C1)NCC1CCCN(C(c2c(C)cnnc2O)=O)C1 C1(CC(=O)N(CCN(C(C23C(CN(C(C)=O)C2)C3)=O)C)C)CCC12CCOCC2 c1(CSC)cc(C(=O)NCC2(NC(=O)CCC=CBr)CCCCC2)ccc1F c1(C(=O)NCC(C)NC(C(CCSC)O)=O)cc(F)cc2ccoc12 CCCC(C(N)=O)NC(c1ccoc1CNC(c1ccccn1)=O)=O c1(OC)ccc(OC)c(CC(=O)NC(C2CN(C(=O)CCc3ccon3)C2)C)c1 N1(C(C(n2c(C)ncc2)C)=O)CC2CC2(CNC(c2c[nH]c(C(=O)OC)c2)=O)C1 c1(COCC(=O)NC(C)CNC(=O)CSc2ccccc2)ccnc(O)c1 C12(CNC(CCCOCC=C)=O)CC(CN1C(=O)C(C)(C)F)C2 C1(CC(N2CC(Cn3cc(CC(C)O)nn3)C2)=O)CCC(F)(F)CC1 c1(C(N2CCOCC(NC(C(C)C3CC3)=O)C2)=O)cc2cc(F)ccc2[nH]1 c1(C(N(C2CCCN(C(C3(C4CC4)CC3)=O)C2)C)=O)cccc2c1NCC2 C1(CC)CN(C(=O)CNC(=O)C(F)(F)F)CC1(F)C(=O)Oc1ccccc1SC c1(OC)cc(N)c(F)cc1C(=O)NC1(C)CC(NC(c2ccoc2)=O)C1 C(C)(C)(CC(=O)NCC1CN(C(c2cnns2)=O)CC1C)OC Cc1c(CN2CCC(NC(=O)C(F)(F)c3ccccc3)C(F)C2)ccnc1Cl c1(OC)cc(C)ccc1C(=O)NC1CCCC1NC(=O)CC1CC1C(F)(F)F C1(C(=O)NCCCCn2cc(-c3c(SC)cccc3)nn2)COC2COCC12 c1(C(=O)NCC2C(CC)CCN2C(=O)Cc2ccsc2C)cc(C)c(F)c(C)c1 C1(C)(C(N(CCCNC(C=CC(=O)N(C)C)=O)C(=O)C2CC2)=O)CCCNC1=O C1(C)(CC)CCC(C(=O)NC2(CNC(=O)C(=Cc3ccccc3)C)CCCC2)O1 c1(C(=O)NC(CN(C(=O)CC2CC3C=CC2C3)CC)C)cccc(C)c1 CC1CN(C2CC2)CC1NC(=O)Cn1cc(CNC(C2(C)SCCCS2)=O)nn1 N1(C(c2cccc(OC(C)=O)n2)=O)CCC2(CCN(C(c3cc[nH]n3)=O)CC2)C1 CC(C)(CO)CCNC(C1CC(=O)CN1C(C1COCC1(C)C)=O)=O C1(C(N(C2CCN(C(=O)CC(CC)SC)C2)CC#C)=O)CCCCC1CC CC1CC(=O)NCCN1C(=O)COC1CCN(C(c2cc(O)cc(=O)o2)=O)C1C c1(C(N2CC(C)N(c3ncc4ccsc4n3)CC2)=O)ncnc2ccc(Br)cc12 N1(C(C2CCC(C)CC2)=O)Cc2occ(C(=O)NCCC3CC3C)c2C1 C(N=c1[nH]cnc2ccsc12)C1N(C(c2c3ccc(OC)cc3[nH]c2)=O)CCC1 C1(OC)CN(C(C2C(C#N)C2(C)C)=O)CC1NC(=O)C(F)(F)c1cnccn1 c1(C(N(CC)CC2CCCN2C(C2CC2C)=O)=O)cccc2ncc(C)cc12 CC(C(=O)NCCN(C(=O)COCC(F)(F)F)C1CC1)=CC1CC1 N1(C(CC(CCOC)(C)C)=O)CCCC12CCN(C(=O)CC1(C)CCOC1)C2 CC1CCCC=C1C(=O)NCC1C2CCC(C2)N1C(c1coc(CC2CC2)n1)=O C1(CC(N2CCC(N(C(=O)C(F)=CC3CC3)CCC)C2)=O)CC(C)(C)OC1=O c1(CCCC(=O)N2CCCC2Cn2cc(-c3ccns3)nn2)ccc(Cl)cc1 C(=O)(C(F)CC(CC)CC)NCc1occ(C(=O)NC(C(CC)C)CO)c1 CN=c1[nH]c(=NCc2cc(Br)cs2)[nH]c(=NC(C)Cc2ccco2)[nH]1 c1(N2CC=CC(NC(C(C(CC)O)(F)F)=O)C2)nc2cccc(F)c2cc1C#N C1(C)(NC(CC(=O)OCC)=O)CCCCC1C(=O)NCc1cccc(O)c1C.OCC N1(C(=O)C#CC2CCCCO2)CCCC2(C1)CN(C(=O)C(F)(F)C1CC1)CCO2 N1(CC(N2CCCC(c3[nH]nc(C(C)(C)C)n3)C2)=O)CCCC2CCNCC12 C1(=CC(=O)NC2C3(CC(NC(c4cc(C)oc4C)=O)C3)C2)CN2CCC1CC2 c1(C(C)C)cccc(C(N2CC(C(C)(C)O)(CNC(C3CC(F)(F)C3)=O)C2)=O)n1 C1(C(=O)NCC2(NC(=O)C(c3ccc(F)cc3)=O)CC2)CCC2(CC1)CC2(F)F C1(N(C(=O)C(F)OC)CCCC)CCN(C(=O)Cn2cncn2)CC1 c1(OC)cc(CNC(c2ccc(F)cc2OC)c2nnnn2C(C)C)cc(Br)c1 C1(N(C(C(COCC)NC(=O)C=CCO)=O)C)CCC(=O)N(C)C1 CC(C)CC(C(=O)NCC1(O)CCN(C(C2CCC(C)(O)CC2)=O)C1)N(C)C C12(C(=O)NCC3C(NC(c4c(COC)ccs4)=O)C3)COC(CF)(C1)C2 c1(SCC(N2CC(CCNC(C(CC)(C)O)=O)OCC2)=O)cc(C)ccc1C C1(NC(C2CC(CC)(CC)C2)=O)CC2CC(C1)N(C(c1ccc(Cl)c(O)c1)=O)C2 C=CCCCC(=O)NCCCCC(C)NC(c1ccc(C(N)=O)s1)=O c1(N(CC(C2CCCC2)OC)C)nc(=N)[nH]c(=NC(C)CC2CCCO2)[nH]1 C1(C(N2C(C)CC2(C)C)=O)CCN(C(=O)C2CCOC(=O)CC2)O1 c1(NC(C(C(C)CSC)N2CCC(=Cc3cccs3)CC2)=O)ccc(Br)c(F)c1F CC1CCCC=C1C(=O)N1CCCC1(C)C(N1CC(=O)NC(=O)C1C)=O c1(NC(COCCOCCOC)=O)ccc(Cl)cc1NC(C1(CN)CCCC1)=O.OC C1(NC(C2(C=C)CCC2)=O)CC2CC1N(C(C1CCC(F)(F)C1)=O)C2 N1(C(C(C)(C)F)=O)CCC2(CCCCC2NC(C2CC2C(N)=O)=O)CC1 C1(F)(CNC(C2N(C)CCOC2)=O)CCN(C(=O)COCC2CCOC2)CC1 Cc1c(C(=O)NCC2CC(NC(=O)C(C3CCOCC3)C)C2)sc2ccccc12 c1(OCCN(CC)CC)ccc(OC(C)C(=O)N(C)CCCC)cc1 N1(C(c2nccnc2Cl)=O)CC(C2CCCCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 CC1CN(C(C2COC(=O)N2C)=O)CCN1C(C1CCCNS1(=O)=O)=O C1(C(=O)NCC2(CC)CC(CO)C2)C(CC)CCCN1C(=O)C1=CC(C)(C)C1 C1(NC(CCc2nc(C)sc2)=O)CCC(Nc2ncc(I)cn2)CC1 C1(CNC(C2(CC#C)CC=CCC2)=O)COC(C)(C)CN1C(c1csc(Cl)c1)=O N1(C(CSC)=O)CC(NC(c2cnc(C(C)C)nc2)=O)C2CCCC2C1 CC(C)(CC(=O)N1CCCC2C1CCN2C(=O)CCCS(N)(=O)=O)CC(F)(F)F C12(C(=O)NCC34CCN(CC3)C4)COCC1CN(Cc1nsc3ccccc13)C2 N1(C(c2nc(C)c(C)[nH]2)=O)CCC(NC(=O)CCNC(=O)CC(C)C)C(F)C1 N1(CC)CCCC(ONC(=O)C(C)NC(=O)C(Cn2cccn2)N(C)C)C1 CC1CC(NC(=O)Cc2cnccn2)CCN1C(=O)Cc1nccs1 C1(NC(CN(C(C)=O)C)=O)CCC2CN(C(c3cn(C(C)C)nn3)=O)CCC2C1 N1(C(C2CCC(n3cc(C4(O)CC4)nn3)C2)=O)CCC(O)CC12CC2 C1(CCOC)(NC(=O)CSc2ccccn2)CCN(C(C2(C#N)CC2)=O)C1 C1(c2n(C)ccn2)CC(C(=O)Nc2ncccc2Cl)NC(=O)N1 C(=O)(CS(=O)(=O)NC)NC1CC(NC(CN(C(=O)OC)C)=O)C1 C(=O)(C(F)(F)c1nccs1)NC1(CN(C)C(C2(C)CC2(F)F)=O)CC1 CC(C(F)C(=O)NCCN(C(C(=O)Nc1ccc(Cl)c(F)c1)=O)C)C(F)(F)F C1(N(C(C(CC)OC)=O)C)CCCN(C(=O)C(F)(F)c2ccccc2)C1 C1(C(=O)NCC2CCCC(=O)N2)(CNC(=O)Cc2nnc(O)o2)CC12CCC2 N1(c2nc(N(CC(C)(C)OC)C)nc3c2n(C)cn3)CCc2c(Cl)cccc2C1 C1(C(=O)NC2CCCN(C(C3C(C)C3)=O)CC2)CCc2cc(F)ccc2O1 N1(C(CC2(COC)CC2)=O)CCC2CN(C(c3cc(Cl)ns3)=O)CCC2C1 C12CC3CC1CC3C(=O)N2.C(C)(C(=O)N1CCC(N(C)C)C1)(C1(C)CC1)OC CCC(CO)C(=O)N1CCOC(C(C)NC(=O)CCN2CCCCC2)C1 C(=O)(CCCS(N)(=O)=O)NC1CCCN(C(CCSCC)=O)C1C C1(NC(CCCCCSC)=O)CC2CC(C1)N(C(c1cnn3c1OCC3)=O)C2 CCCCCCCC(=O)NCC(F)(C(=O)N(C1CC1(C)C(F)F)CC)C(C)C N1(CC(=O)N(C)CC2N(C(C3C(C)C3)=O)CCC2)CCCNS1(=O)=O C1(CN(C)C(c2ocnc2C(F)(F)F)=O)CN(C(=O)CC2CCCO2)CCO1 C1(C(=O)NC2(CO)CCCC2)COC2(CCN(C(=O)Cc3ccc(F)nc3)C2)C1 N1(c2nc(COC)nc(N3CCC(OC(C)=O)CC3)c2)CC2CCC(CO)(C2)C1 CCCC(C(=O)OC)C(=O)N1CCOCCC1C(=O)NCC1=NOC(C)C1 c1(CNC(COCCC(C)C)=O)cc(O)nc(CNC(C2COC(C)(C)C2)=O)n1 CC1(C)C(NC(c2ccn(C3CC3)n2)=O)CC1CNC(c1cc(F)c[nH]1)=O C(=O)(C(CO)C(C)(C)C)N1C2CC(CNC(c3c(C)c(Cl)ccn3)=O)(OC2)C1 c1(C(N(C)CC2(NC(=O)CCn3cnnn3)CC2)=O)ccn2cccc2c1 c1(C(=O)NCc2c(CNC(CC(C)OC)=O)cccc2)ccc([N+](=O)[O-])cc1 C1(C(=O)NC2C(C(=O)NCCc3ncco3)CC2)CCCC12CC2 C(=O)(C1=CC2(CCOCC2)C1)NCC1C2CN(C(C(CCCOC)C)=O)CC21 Cc1ccc(CN2CCC(C(=O)Nc3ccc(C#N)cc3F)C2)c2ccccc12 C1(CC(N2C(CNC(c3c(C)cc(CC)o3)=O)CC2)=O)COc2ccccc2O1 CC1=C(C)CC(C(N2CC(F)CC2CC(=O)NC(c2cccs2)C)=O)CC1 c1(C(=O)NCC2(F)CC(NC(=O)C(O)C3CCC3)C2)cnc2n(c1=O)CCS2 c1(OC)cc(CCC(=O)NCc2cn(CC(C)NC(C)=O)nn2)cc(Br)c1OC C1(CNC(=O)CC2CC23CC3)CN(C(=O)CCF)CCO1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(CC#C)CC(=O)Nc1ccc(Cl)nc1 c1(C(=O)NC(CCNC(Cc2c(C)cco2)=O)C)nc2ncc(CCO)cn2n1 C=CCC(C(=O)NC(C)(CNC(c1cncc(CC)c1)=O)CO)N(C)C CS(=O)(=O)C(CNC(c1cc2sccc2s1)=O)CNC(C12CC(F)C1C2)=O Cc1ccc2c(c1)CC(C(N1CC=CC(NC(=O)CNC(=O)C(C)(C)C)C1)=O)S2 n1(CC(=O)NC2CCN(C(Cc3nc(C)sc3Cl)=O)C2)nc(C)c(C)c1C N1(c2cc(OC)ncn2)CCC(NC(=O)CC(C)CN(C)C)C2(CCC2)C1 CC1(CNC(=NCCOC(F)(F)F)NCC(F)F)CCC(F)(F)C1 c1(CNC(=O)N(C2CCC(=O)NC2=O)CCO)ccc2c(c1)CCC2 c1(CCC)nsc(N2CCC(NC(c3cn(C4CCCCC4)cn3)=O)C2)n1 C1(NC(CN(CCC)C)=O)CCC(C)(C)CC1CNC(c1ncnn1CC)=O Cc1cc(C(N2CCCCC2CCNC(c2ncsc2C(C)C)=O)=O)oc1C Cc1nc(S)sc1CC(=O)N(C(C)CCNC(=O)C(C)OC1CCCC1)C C(=O)(C(CN(C)CC=C)c1ccccc1)NCCN(C(CC=CC=C)=O)CCC C(CCCCN=c1nc2c(cnn2C)c(NCCC2OCCC2(C)C)[nH]1)OC c1(N2CC(CC)OCCC2)ncnc2c1ncn2CC1(CC)CCOC1 S(=O)(=O)(c1ccc2c(c1)CC(C)(C)O2)NC(c1nnnn1CCCF)(CSC)C c1(CNC(C2(OC)CCC2)=O)nc(CNC(C2CC2(F)Cl)=O)cc(O)n1 Cc1cc(N(CCCN(C(=O)CC(C)(C)O)C)C)nc(-c2cccs2)n1 N1(CC(C)NC(=O)OC(C)(C)C)CCOCC12CCC2.c12cccc(c1)C(=O)N2CCl CC#CCCCC(=O)N1CCC(CC(C)NC(C2CCC2OCC)=O)CC1 C(CCCCCC(=O)N1CCCC1CCCNC(C1(C(C)C)CC1)=O)SC O=C1NCN(CC(C2CCCCC2)O)CCc2ccsc21 O=C(CCCc1nc(-c2ccccc2)no1)NC1CN(C(=O)COCCCF)C1 C1(=O)C(CCc2ccccc2F)N1C.C(CS(C)(=O)=O)N(C(C)C(=O)OC)CC=C c1(OC)nc(Cl)cc(=NC(=O)c2sc(=NCc3cc(F)c(F)cc3Br)[nH]c2C)[nH]1 C1(C(N2CCC(CNC(c3occc3CO)=O)C(C)C2)=O)(OC)CCCCCC1 c1(CC(=O)NC2C=CCN(C(c3c(Cl)cc(C)s3)=O)C2)cn2c(C)csc2n1 C1(CC(=O)Nc2ccc(F)nc2)CC2(C1)CN(C(=O)C=CC1CCOCC1)C2 N1(C(c2cncc(C)c2)=O)CCC(C)(CC(=O)NCC2(CO)CC2(C)C)CC1 N1(C(C(CC)=CC)=O)CC(OC)C(NC(c2cnc(CC(C)C)[nH]2)=O)C1 c1(CC(N2C3CCN(C(C(COC)(C)C)=O)C3CC2)=O)c[nH]c2cc(Cl)ccc12 c1(C(=O)NCC2(F)CC(NC(c3cc(C#N)oc3)=O)C2)n[nH]c2c1CCC2 C1(CC)CN(C(=O)CC2CCCC(O)C2)CCC1NC(=O)CCNC(N)=O c1(OC)ccccc1CC(=O)NC1CCC(CNC(C2CCC(CO)CC2)=O)C1 C1(NC(c2cc(C3CCC3)no2)=O)CN(C(C2SCCCS2)=O)CCC1O N(C=CC(=O)C(F)(F)F)C(CSC(C)=O)=O.N12CCOC(C1)CC2=O C1(C(=O)NC(C)CC2CCC2)CC12CCN(C(=O)Cc1cncn1C)CC2 N1(C(c2cn(C)nc2Br)=O)CCCN(C(=O)CC2CC2(C)C)CC1 C(=O)(C(C)(CC)CC=C)NC1C=CC(NC(COCCOCC#C)=O)C1 N1(C(c2cnc(Cl)s2)=O)CCCCC1C1CCCCC1 c1(C(=O)NCCC(=O)NC2CCc3ccccc3C2)cncc2nccnc12 N1(C(Cn2ccc(C)n2)=O)CCC(O)(CNC(C2CC3CC3C2)=O)CC1 C1(NC(C(C)=CC)=O)CC2CC(NC(=O)Cc3cc(Cl)cc4c3OCC4)CC2C1 c1(OCC)cccc(C(=O)NC(C2CCCC2)CNC(=O)C(C)n2cccn2)c1 N1(C(C=CSC)=O)CC(CNC(C2(CO)CC(C)(C)C2)=O)C2(CCC2)C1 N1(C(C(CC)CC)=O)CC2CN(C(c3ccc(O)cc3O)=O)CC12 C=C1CN2C(=O)CCC2(C(N2CCN(CCN(C(=O)COCCF)C)CC2)=O)C1 CC(C)CCC(O)C(=O)N1CCC(CNC(c2cc(=O)c(O)c[nH]2)=O)C(O)C1 Cc1c(F)ccc(-c2ccccc2CN(C(Cc2cccc(Br)c2)CO)C)c1O N1(C(c2n(CC)ccc2)=O)CCCCC2(CCN(c3nnn(C)n3)C2)C1 C1(C)(C(=O)NC(c2nc[nH]n2)CC)CCN(C(=O)CC2CC(C)=NO2)C1 c1(-c2n(-c3cccc(OCC)c3)nc(CCOC)n2)cnc2[nH]cnc2c1 N1(C(CSC)=O)CCN(CCN(C)C(c2nnsc2C2OCCO2)=O)CC1 C1(CC(=O)NCc2cc(C(=O)NC3(C)CC4(CC4)C3)no2)CCC2(CCC2)O1 CC(C)(CC(=O)N1CC2C(NC(c3cc(C4CC4)on3)=O)C2C1)C1CCCCC1 c1(SC)cc(C(=O)N(C)CC2CCCC2(C)C)ccn1 c1(OCC=C)cccnc1C(N1CCCCC1CNC(=O)CCCOC)=O CC=C=CCCN=C(NCc1cc(C)cc(Cl)n1)NC1CCCS(=O)(=O)C1 c1(CNC(=O)NC2(C)CC(NC(=O)OC(C)(C)C)C2)ccc(N)c(C)c1F N1(C(CCC(=O)OC)=O)CCCC2(C1)CN(C(=O)COC(F)(F)F)CCO2 N1(C(C(F)OC)=O)CC(CNC(=O)CCC2CCCC2)C(n2ccnn2)C1 CC1CCC(C)(C(=O)N(C)CCN(C(=O)C(C)n2cccn2)C(C)C)C1(C)C c1(C(N2CC(NC(CCS(N)(=O)=O)=O)C(C(F)(F)F)C2)=O)ccc2c(c1)CCC2 c12cc([nH]n1)CNC2=O.CC(CCN(C(=O)CNC(c1cccs1)=O)C)O.CO C1(CCNC(C2CCSC2)=O)CCN(C(c2cc(-c3ccco3)[nH]n2)=O)CC1 C(c1cccnc1)=CC(=O)NCC(C)CNC(=O)C(C)(O)c1ccccn1 C1(C(N2CC(OC)CC(OC)C2)=O)CN(C(=O)C=C(C)C(F)F)C2(CCC2)C1 c1(CC(=O)NC2(C)CN(c3snc(CCC)n3)C2)ccc2nsnc2c1 Cc1cc(C(=O)NCC(C2CCCCC2)NC(C2COC(C)C2)=O)c[nH]1 C(C(=O)NCc1ccc(C(=O)NC(C)CN2CCOCC2)s1)(C(C)C)SC c1(CC(=O)NC(CNC(C(C=CC)O)=O)C(C)C)ccc(Cl)cn1 c1(N(CC(N2CCN(C(N)=O)CC2)=O)C)ccccc1NC(=O)OC(C)(C)C C(=O)(CC(=O)N(CC)CC1(F)CN(C(=O)C(O)Cc2cnc[nH]2)C1)NCC#C N1(C(C2(F)CCN(C(CCN=[N+]=[N-])=O)C2)=O)CCN2CC(F)CC2C1 C1(CC(N2CCCC(CN3CCC(N)CC3)C2)=O)CC2(CCOCC2)C1 N1(C(CC=C)=O)CCCCC1CCN(C)C(c1cn(C)nc1Cl)=O C(c1cnccc1C)=CC(=O)NCC1(CNC(CCC(C)SC)=O)CCCCC1 CCC(CC)CC(F)C(=O)N(C1CCN(C(C2(F)CC=CC2)=O)CC1)C S(=O)(=O)(c1cn(C)cn1)NCC(N1CCC(NC(C(F)=C(C)C)=O)C(C)C1)=O c1(C(N2CCn3ncc(CNC(C4(Cl)CC4)=O)c3C2)=O)cc2cc(F)ccc2o1 C1(CCSC)CCN(Cc2cnn3c2CN(C(=O)C(N)=O)CC3)CCC1(F)F C1(NC(c2ccc(C#C)o2)=O)(CNC(=O)COC2CC=CC2)CCC(F)(F)CC1 C1(NC(C2CCC(=C)CC2)=O)COCCN(C(c2cnc(C(N)=O)s2)=O)C1 c1(CC)ccc(CNC(=O)CCc2csc(C)n2)cc1.C12CCCC1C(=O)NC2 C=CCC(C(=O)N1CCC=C(F)C1)NC(c1cccc(CC)n1)=O N1(C(c2nc(C)[nH]n2)=O)CCOCC(NC(c2ccc(O)nc2Cl)=O)C1 C1(C(N2CCC(C(C)(C)NC(c3c(C#C)c[nH]n3)=O)C2)=O)CC2CCC(C1)N2C Cc1cc(C)n(CCC(=O)NCC(C)(C2CC2)NC(C2CC2[N+](=O)[O-])=O)n1 C1(O)(C(N(CCN(C(=O)C(c2ccccc2)O)C)C)=O)CCN(C(C2CCC2)=O)C1 c1(CNC(C(n2cc(-c3ccc(F)cn3)nn2)C)=O)ccc(N)cc1F CC1(C)CN(Cc2ccc(O)c(F)c2)CCC1NC(c1ccncc1F)=O CC(C)(CNC(C1CCC(C2CC2)C1)=O)CC(=O)NC1CCCC1CF Cn1cc(C(=O)NC2CN(C(c3cnn(C)c3Cl)=O)C3CC23)c(C(F)F)n1 C(=O)(C1=CC(C)(C)C1)NCCC(CNC(c1ncc(OC)nc1)=O)O C1(CCC(=O)NC2(C3N(C(CCC4C(C)(C)C4)=O)CCC3)CC2)CCCCCC1 c1(CNC(C2CC(C)CN2Cc2ccc(O)cc2)=O)ccc2c(c1)OCO2 C1(O)(CC(=O)NCC2N(C(CCNC(C)=O)=O)CCC2C)CCCN(C)C1 CC1CN(C(C2(n3cccn3)CC2)=O)C(C)CN1C(=O)CC(C)C(F)(F)F N1(C(C2CC(CC)C2)=O)CCC(CNC(C2CCCN2C2CCCC2)=O)C1 N1(C(CN(CCC)C)=O)CCC(N(C2(c3ccc(C)cc3)CC2)C)CC1.C1CO1 N#Cc1ccsc1C(N1CCCC(CCNC(C2CCOC2C2CC2)=O)C1)=O c1(SC)cc(C(=O)Nc2c(Cl)cc(C)cc2Cl)cc(SC)c1 Cc1ccc(C(F)C(N2CC(NC(=O)CN3CC(C)(C)C3)C(C)C2)=O)cc1 c1(C(=O)NC(C)C(=O)NC(C)(C)C(=O)N(C)C)ccc2[nH]nc(Cl)c2c1 N1(C(CCCOCCC)=O)CCC(C)(C(=O)NCc2coc(C)c2)C1 C=CCCC(=O)NC1CCN(CCCOC(C)=O)C1.C12CC(C1)NC2=O.OCC CCCCS(=O)(=O)CC(=O)N(CCCNC(=O)CCc1cnc2n1CCCC2)C CC1(C(N2CC(NC(c3cscc3Cl)=O)C(O)C2)=O)CCNC(=O)C1 c1(C(N2CCC(NC(C(C(=O)OCC)F)=O)CC2C)=O)c[nH]c2cccc(C)c12 C1(CC(=O)NCC(CCCC)O)CN(C(=O)CC=C(C)C)CC12CC2 N1(C(C=CC(CC)=CC)=O)CC(NC(c2c[nH]nc2CC)=O)CC12CCOC2 C1(CNC(C(C)(C)F)=O)CCC2CN(C(=O)C(c3ccccc3)O)CCC2C1 Cc1cccc2sc(C(=O)NCCOCCN(C(C)C(=O)NC3CCC3)C)c(Cl)c12 c1(C(=O)NC2(CNC(CC)=O)CCOC2)cc(C)oc1C C(=O)(C(C)(C)CC(F)F)N1CCC(CNC(CNC(c2cc(C)nn2C)=O)=O)C1 N1(C(c2cc(C(C)=O)sc2)=O)CC(NC(=O)C(O)CF)CCC1C C1(NC(=O)COCCO)CCN(C(C2CC3(CCOCC3)CO2)=O)C12CCCC2 c1(OC)ccc(C(C)=CC(=O)NCC(C)NC(c2cc3sccc3[nH]2)=O)cc1N C1(NC(CCC(C)SC)=O)COCCN(C(=O)CSc2ccc(O)cc2)C1 c1(NC(C)C)cccc(C(N2CCC(NC(=O)COC3CCOC3)CC2)=O)c1 c1(C(=O)NC23CCN(C(CC4(C)CC4)=O)CC2C3)ccc2nc(S)oc2c1 C1(C)(NC(c2nc(CNC(c3c(C)nco3)=O)oc2)=O)CC(C)(C)OC1=O c1(C(=O)NC2C(NC(C=CC)=O)CCOC2)cc2ccncc2c(O)n1 C(CNC(c1cc2n(n1)CCC2)=O)(C(C)C(C)C)NC(c1cc(OC)n(C)n1)=O C(=O)(C(C(C)C1CCCCC1)N(CCC)Cc1ccc(Cl)cc1)NCCC Cc1cc(NNC(=O)Nc2ccc(C(F)(F)F)cc2Cl)ccc1Cl Cn1ccc2ccnc(C(=O)NCCCCCNC(=O)C#CC3(C)COC3)c12 N1(C(C2C(c3n(C)cnc3)OCC2)=O)CC2CC1CN2C(c1ccc(CO)o1)=O O=S(=O)(c1ccc(Br)cc1NCCC1CC1(Cl)Cl)N1CCCC(NCCO)C1 C(=O)(CC(O)CNC(c1nccn1CC)=O)NCCN(C(CC)C)C CC(C)C(O)CC(=O)N1CC2(CCC2NC(=O)C=Cc2ccc(Br)o2)C1 c1(CC)ncccc1C(=O)NC1CCCN(C(=O)CC2C=CCCC2)C1 c1(OCC(N2CCCC(CCNC(C(CCC)O)=O)C2)=O)ccc(Cl)cc1Cl c1(NC)cnccc1C(=O)NCc1cc(C(=O)N(C(C)C(C)C)C2CC2)ccn1 N1(CC(=O)NCCC2(O)CCCN(C(CC(C)C)=O)C2)CCCCCCC1=O CC(C)C(F)C(=O)N1CCCC1(C)CNC(=O)C=Cc1ccoc1 CC1CCC(C(=O)NCCOCCOCCCNC(c2nonc2N)=O)C1 C1(C(=O)NCC(C)N(C(c2nc(C)sc2)=O)C)Cc2nn(C)cc2C(=O)N1 CC1CN(C(=O)C(c2ccc(Br)s2)C)CCN1C(c1ccn(C(F)F)n1)=O CC1CCN(C(C23CC(CO2)C3)=O)CCN1C(C1CC2CC1C1CC21)=O CN1C(=O)N(C2CC(c3cc(I)ccc3F)C2)C(=O)C1=O C1(NC(c2cccnc2)=O)C2CC1CN(C(c1cc(C(F)F)ccn1)=O)C2 Cc1c(C(=O)NCCC2CCCCNC2)cccc1-n1cnnc1 C1(CNC(C2(C)ON=C(C)C2)=O)CC2(CC2)CN1C(c1ccncc1O)=O C=CCC(C)(CNC(C1(N(C(=O)C(C)OC)C)CC1)=O)CO N1(C(C2CC(SC)C2)=O)CC(NC(=O)C(n2ccnc2C)C)C(F)C1 N1(C(c2cccc(OC)c2)C(=O)NC2(C)CC2)CC2CC3CC(C2)CC1C3 CCC(C)(O)Cc1cn(C(C)C(=O)NC(C2(OC)CC2)C)nn1 N1(C(=O)OC(C)C)CCC(NC(=O)NC2(CCCF)CC2)CC(O)C1 N1(C(c2cncc(SC)c2)=O)CCCC(C)(CNC(C2CCC(=O)NC2)=O)C1 c1(C(=O)NCC2C(NC(Cc3n(C)cnc3)=O)CC2)cccc2c[nH]nc12 C1(C(=O)NC(CC)C2CCC2)CN(C(C2COCOC2)=O)CC1C1CC1 c1(OC)ccc(C(N2CCC(NC(c3ncccc3CSC)=O)C2C)=O)cn1 C(=O)(C1CCCc2nc[nH]c21)NCC1N(C(C2(CCCC)CCC2)=O)CC(O)C1 N1(C(C(C2CCCC2)OC)=O)CCC(C)(C)C1CNC(c1cc(C2CC2)no1)=O C1(CNC(C(C)(C)OCC)=O)CCCN(C(C2(CO)CCOCC2)=O)C1 c1(C(=O)NCC(C)NC(C2CC(SC)C2)=O)cccc(Br)c1 C1(NC(C(F)=CCC)=O)CN(C(=O)CCc2ccncn2)CCC1C CC1CN(C(c2[nH]nnc2-c2ccnn2C)=O)CCC1NC(c1cc(Cl)c[nH]1)=O CCC(C)CC(C)C(=O)N1CC(CO)C2(C1)CN(C(C1CSCCS1)=O)C2 c1(OC)cccc(S(=O)(=O)N(CC(c2ccc(Cl)c(Cl)c2)O)C)c1OC CC(=O)CCCC(C)(C)C(=O)N1CCC(NC(c2cn(C)nc2C)=O)C(C)(C)C1 C(C1c2ccsc2CCN1C(C1CC=CCO1)=O)NC(=O)CCc1ccoc1 C(=O)(C1=NOC(C)(C)C1)N1C(C2(C(=O)Nc3cc(C)c(C)nc3)CC2)CCC1 c1(C(=O)NCC2OCC(CNC(C3C(C)(COC)C3)=O)C2)nnc2n1CCOC2 C12(C(=O)NC(CCC(=O)OC)C)CC(CN(C(=O)CCC(C)CN(C)C)C1)C2 C(=O)(C(CNC(C1CCC(=O)N1C)=O)C(C)C)NC1CN(CCC)C1 N1(C(COCCCC)=O)Cc2[nH]nc(C(N3CC(S(C)(=O)=O)C3)=O)c2C1 Cc1cc(C(=O)C(=O)NCC2CCCN(C(=O)CSCCC(C)C)C2)ccc1F c1(C(=O)NCC(CC)NC(=O)C(C)C2(O)CCC2)cccc2c1ncn2C c1(C(N2CC(C)(CC(=O)OC)C2)=O)cnc(N)c(Cl)c1.C1(=O)CCCN1 N1(C(C)=O)CCC2(CCCC2NC(=O)NC2CCC(C3CCC3)CC2)CC1 n1(CCC)nc(C)c(C(N2CCC(O)(CNC(=O)C(O)C(C)(C)C)C2)=O)c1C C1(C(N(CC)CC2(OC)CCOC2)=O)CCC(C)(C)N(C(=O)C(C)(C)Cl)C1 CC1(C)COCC(CC(=O)NCC2CN(C(=O)Cc3ccoc3)CCO2)O1 N#Cc1ncccc1-c1cncc(C(=O)Nc2cnc(F)c(Br)c2)n1 CC1CN(C(=O)C=Cc2cocn2)CC1NC(=O)C(=O)Nc1ccccc1CO n1(CC)nc(C(=O)NCCC2CC(NC(C3(C)CC3F)=O)C2)c(C)n1 c1(CNC2CC(C(C3CC3)Nc3c(C)n(C)nc3)C2)cc(O)c(O)cc1O N1(C(C(CNC(COCCCC(C)C)=O)O)=O)CC(=O)N2CCCC2C1 C(CCCCC(=O)NC1CCCCC1NC(=O)CNC(=O)Cn1cncn1)=CC CCC(C(=O)NC1CCC(CCNC(C2CC(=O)C2C)=O)C1)OC c1(C(=O)NCC(CC)N(C)C(C2CC3(CC3)CN2C)=O)cc(C)n(C)c1C N1(C(CNC(CC)=O)=O)CCCC(C)(C)C1CNC(c1cscc1OC)=O C1(C(c2n(C)nnn2)(C)Nc2ccccc2P(C)(C)=O)C2CC3CC(C2)CC1C3 N1(C(C(CC2CC2)OC)=O)CC(C)C(C)(CNC(C2(C)SCCCS2)=O)C1 C1(NC(C=CCOC)=O)CCn2ccnc2C1.c1(CC2C(=O)N2)cnn(C)c1O C(c1ccco1)=C(C)C(=O)NCC1C=CCN1C(=O)COCCCF C(=O)(CCCS(C)(=O)=O)NCC(CNC(=O)C=CC(C)(C)SC)OC c1(N2CC(CCNC(c3cc(C)ccc3Cl)=O)(OC)C2)ncc2c(n1)CCOC2 C1(CCN(C(C(C)C2C(C)C2)=O)C2CC2)CCCCC1 C1(NC(=O)CCc2cscn2)CC2CC(C1)N(C(c1ccc(Cl)nc1Cl)=O)C2 C=CC1(CC(=O)NCC(C)(CC)NC(C2CC(N3CCOCC3)C2)=O)CCC1 c1(COC)ccc(C(=O)NC(CNC(=O)COCc2ncnn2C)CO)s1 c1(C(C(=O)NC(C)(C)C)N(CCCF)C)cc(-c2ccccc2)on1 CCC(CC)CCCC(=O)NC1(C(=O)NOCC(=O)OCC)CCSC1 C1(NC(C2(CC(C)=O)CC2)=O)CC(C)(CNC(=O)Cc2cnc(C)s2)C1 C1(NC(COCCOC)=O)COC2(C1)CN(C(c1scnc1Cl)=O)C2 c1(C(N(CCN(C(c2c(CC)nn[nH]2)=O)C)C)=O)ccc(C2CCC2)nc1 C(c1ccco1)=C(C)C(=O)NCC1CCCN1C(C1CC(CC(F)(F)F)C1)=O C1(CNC(C(C)O)=O)CCN(C(c2cnccc2C2OCCO2)=O)CC1(F)F c1(C(=O)OCC(COC)O)ccc2cccc(Cc3ccc(OC)cc3)c2c1 Cc1[nH]nc(C(N2CC3CC2C3C(=O)N(CC(C)(CO)N(C)C)C)=O)c1O N1(C(C(CC)COC)=O)C(C)CC2CN(C(c3c(C)sc(C)c3C#N)=O)CC12 c1(OC)cnc(CNC(C2(NC(c3cn(C)cc3C)=O)CCSC2)=O)cn1 c1(CCC(=O)NC2C(NC(CN(C)C)=O)CCCC2)ccc2c(c1)OCO2 N1(C(c2c(C)onc2Cl)=O)C2CCC1CN(C(c1cc(C)n(C)n1)=O)CC2 c1(N)nc(Cl)nc2c1CCCC2.N1(Cc2cn(CC)nn2)CCC2(COC(C)C2)C1 C1(C(=O)NCCCCNC(=O)C(F)CC2CCC2)CCC2C(C1)C2(F)F c1(OC)ccc(F)c(C(=O)NCC2CCCCCN2C(C2(OC)CCC2)=O)n1 c1(C2(C(=O)NC3(C(=O)O)CCNC3)CC2)ccc2c(c1)OCO2 N=c1cc(C(=O)Nc2ccc(C34CCC(C(=O)OC(C)(C)C)(C3)C4)cc2)cc[nH]1 C1(N(C(=O)CC2(SC)CC2)CC#C)CCN(C(=O)CNC(=O)OC(C)(C)C)C1 C#Cc1ccc(CC(N)C(=O)NC2CC(NC(N)=O)C2)cc1 C1(C(=O)NCCc2c(C)nccn2)COCCN(C(C2CC=CCC2C)=O)C1 CCCCCC(O)CC(=O)N1CC=C(C(N2CCNC(=O)CC2C)=O)C1 C(=O)(CS(=O)(=O)Cc1ccccn1)N(C)CC1(NC(c2cn(C)cn2)=O)CC1 c1(-c2cc(CCCC)[nH]n2)nc(Cc2ccc(Cl)cc2)nn1CC C1(CN(C)C(c2nc(=O)n(C)[nH]2)=O)CCN(C(C2CC3CCC2C3)=O)CC1 C(CCNC(c1ccc[nH]1)=O)(C(=O)NCCn1ccnc1)OC c1(C(N(C2CN(C(C(CC(C)C)(F)F)=O)C2)C)=O)cc2c(nc1N)CCCC2 c1(OC)c(C)csc1C(=O)NCC1CCC(NC(=O)CCn2c(C)ccc2C)C1 C1(C(N2CCN(C(=O)CC34CCCC3C4)CC2)=O)CC(=C(F)F)C1 C(=O)(CCCC(C)O)Nc1cccc(NC(C(C)NC(=O)NC)=O)c1 c1(C(N(CC(=O)NC(c2ncc(C)[nH]2)CC)CC)=O)cn(C)nn1 O=C(CCC(F)(F)F)NC1CC2CC1CN2C(=O)C(F)(F)c1nccs1 N1(C(C=CC)=O)CC(C(=O)NCC2OCCC2(C)C)CC12CCC2 c1(OC)ccc2c(c1)CCC(C(=O)OC1COC1)C2.c12cccn1c2=O C1(CNC(c2nnn(CC)c2C)=O)COC(C)(C)CN1C(C1CC1CF)=O Cc1cc(Cl)cc(N)c1C(=O)NC(CCN(C(=O)C=Cc1cnc[nH]1)C)C(C)C C=CC(CC)CC(=O)NCC1CC1CC(=O)NCC1CCCCS1 N1(C(COC)=O)CCCCC1CNc1ncc(-c2ccccn2)cn1 c1(CC(=O)NCCN(C(CCCSC)=O)C2CCCC2)cc(F)cc([N+](=O)[O-])c1 C(=O)(CCC(C)(C)c1ccc(F)cc1)C(C)N=c1[nH]c(-c2nn[nH]n2)cs1 c1(CCC(=O)NC2C(NC(C(C)(C)F)=O)C2)cccc(OC(F)(F)F)c1 C=C(C)CC(C(=O)N1CCC(n2cc(-c3ccccc3OC)nn2)CC1)OC c1(C(=O)NCC2(NC(C3N(C)CCC3)=O)CC2)cc(O)cc(N)c1Cl c1(CC(=O)NC(C(C)NC(C2CCS(=O)(=O)C2)=O)CO)ccc2c(c1)CCOC2 C1(F)(C(=O)NCc2n(C)ncc2)CCN(C(=O)CCC2CC2)C1 C(C(=O)NCc1cnn(C)c1C(=O)N(c1ccsc1)CC)(C(C)C)OCC c1(OC)ncc(Br)[nH]c1=NNC(=O)Cc1c(F)cccc1F C(=O)(C1CCCc2nc[nH]c21)N(C(C)C)CCNC(c1cn(C)nn1)=O C12(CNC(=O)C=CCO)CCCC1N(C(C1CC1c1ccoc1)=O)CCC2 N1(C(C(C)CS(C)(=O)=O)=O)CCCC2(C1)CN(C(c1ccc(Cl)nc1)=O)CCO2 c1(CC(=O)NCc2nc(CS(C)(=O)=O)sc2)ccccc1OCC(F)F N1(C(CCC2CC(OC)C2)=O)CCC(C2CC2)C1C(=O)NCC1CCC(C)(C)C1 N1(C(c2ccnc(CO)c2)=O)CCC2(CC1)CN(C(C1CCC=CCCC1)=O)C2 c1(C(=O)NC2C(O)CCN(C(c3c(C)ccc(N)c3)=O)C2)n[nH]c2c1CCSC2 C1(C(=O)NCCC2CCN(C(c3nc(C)n(C)c3C)=O)C2)CN(CP(C)(C)=O)C1 N1(C(C(CC)OC)=O)CC23CCCC2(C1)CN(C(C1CCC2(CCOCC2)O1)=O)C3 c1(C(N2CCC(OC)(CNC(=O)CC3CCCCO3)C2)=O)ccc(C)c(C)c1Cl c1(CC)ccc(CC(=O)NCCOCCN(C)Cc2ncnn2C)cc1F C(C(C)(C)C(=O)N(C)CC1CCCC1NC(C1C2CC3C(C2)C13)=O)SC c1(CN(CC(CC)C)C)cccc(CN2CCOCC2C)c1 O=C(CC1=CCCC1)NCC(CNC(C12CCC(CO)(CC1)C2)=O)CO N1(C(CCOC)=O)CCC(CNC(=O)Cc2sccc2C)(OC)C1 C(=O)(CCCC(=O)C1CC1)N(C)CC1CCN(C(=O)CCc2ccnn2C)C1 C1(NC(c2cc(C)sc2C)=O)CCCC2CN(C(C3CCC(C(N)=O)O3)=O)CC12 N1(C(C2(C)CCOCC2)=O)CCCCC(C(=O)NCC2(F)CC(CO)C2)C1 CCCC(C)(C)CC(=O)NC1COC2C(NC(=O)C(F)(F)CC)COC12 C(=O)(CCC1=NNC(=O)CC1)NCC1CCC(CNC(C2C(C(C)C)C2)=O)CC1 c1(C(N2C(C)CCC(NC(=O)CCCCC3CC3)C2)=O)ccn2ccnc2n1 C1(CC(=O)OC)CN(C)CC1NC(=O)C(C)(C)CN Cc1cccc2cc(C(N3CCCN(C(C4CC(=O)N(C)C4)=O)C(C)C3)=O)nn12 Cc1nc(C(N2CCCN(Cc3noc4c3COCC4)CC2)=O)c2ccccn12 C(=O)(C(C)C(C)(C)C)N(C)CC1N(C(C(CCOC)C)=O)CCCC1 c1(NC(C2N(C(COC)=O)CC(O)C2)=O)c(F)ccc(Br)c1F c1(C(N2C(C3(NC(CC)=O)CC3)CCC2)=O)c[nH]c2ccc(F)cc2c1=O C(C(C)(C)C#CC(=O)NCC1CCC12CCC2)NC(c1ccc(C#C)nc1)=O N1(C(c2ccc(OCC)c(C)c2)=O)CC2(CCCC2NC(=O)CSCC)C1.OCC c1(N(C(C)(C)C)CCOCCO)ccc(F)cc1.c1(CN(CC(O)CO)C)ncc[nH]1 C1(NC(C(C)(C)C2CCC2)=O)CC2(C1)CN(C(=O)CC1CCNC(=O)C1)C2 N1(C(C2CCC(CC)O2)=O)CCC(CC(C)(C)N)CC1 c1(C(=O)NC2CCCC(C(=O)NC(c3ccc(Br)s3)C)C2)ccc(Cl)cc1Br C1(C)(C(N(CCCCNC(c2ccc(-c3cccs3)s2)=O)C)=O)CCNC(=O)C1 C1(CNC(CC2CCN(C(Cc3cc(C)sc3)=O)C2)=O)(CO)CC2CC2C1 C1(NC(CCC=C)=O)CN(C(c2cc(C)c(C)cn2)=O)C(CC)(CC)C1 C(=O)(C(CCC1CC1)Nc1c(C(=O)NC)cn(C)n1)NC1C=CC(C(=O)NC)C1 CC(C)C(C)C(=O)NC1CC(CNC(=O)C(C(C)C)c2ccncc2)C1 C1(C(=O)NCc2ccc(O)c(F)c2)C2CC(O)C(C2)N1C(C1C=CCC1)=O CC1=NOC(C)(CNC(=O)C#CCNC(C2CCCN2C2CC2)=O)C1 N1(C(c2[nH]cc(C#N)c2)=O)CCC2CCC12CNC(=O)CCN1CCCC1=O N1(C(c2ccc(F)cc2)C(=O)N(C(C)C)C2CC2)CCCC(C(=O)NCC(C)C)C1 N1(C(Cc2nc(C)sc2Cl)=O)CCC(CNC(=O)C(F)=C(C)C)C(C)C1 CCC(CC(=O)N1CC=CC1(C)CO)N(C(=O)COC1CCCC1)C Cc1cccc(F)c1C(=O)NCC1CC(NC(C2OCCN(C)C2=O)=O)CCO1 CC(C(C)(O)C(=O)NCCC(C)NC(c1cc2occc2s1)=O)c1ccccc1 CCC(C)(O)C(=O)OC.C1(NC(C2C3C2CNC3=O)=O)C2COCC12 O=S(=O)(c1ccncc1Br)NC1CC2(CCC2)C1 c1(OC)ccc(C(=O)NC2CCN(Cc3nc(C)cs3)C2)cc1 N1(C(CS(CC)=O)=O)CCN(C(c2cc(C(=O)OC)nc(C)c2)=O)CC1C(C)C C1(C)(CC=C(C)C)CN(C(C2CC23CC3c2ccccc2)=O)C1 C(CC1CC1)(C(=O)N1CC(O)(C(C)NC(=O)CCCn2ccnn2)C1)OC C(CC(C)C)(C(=O)N1CCCCCO1)NC(c1c(CC)cc[nH]1)=O N1(C(c2[nH]cc(C)c2C)=O)CCC(NC(C2CC3(CC3)CO2)=O)C1(C)C C1(C(=O)NC2CCCN(C(C)C)C2)(COC)C=CCN1C(=O)C(C)=C1CC1 C12(C(=O)NCCN(C(CC)C)C)CCN(C(c3cc(C#N)cs3)=O)CCC1C2 N1(C(CCc2n(C)cnc2)=O)CCC(CO)(CNC(c2cc(Cl)no2)=O)C1 CCCC(C)CC(=O)N1CC(NC(=O)COCCC(C)C)C(C)(C)C1 c1(C(=O)NC(CCCNC(c2ccc(C(C)C)o2)=O)CO)n[nH]c2c1CCSC2 CCC(C(=O)NCC(O)CNC(=O)C(C)(O)c1ccccc1)OC c1(C(CC)=O)ccc(C(N2CCN(C(C3CCC(C)O3)=O)CC2)=O)cc1 C1(NC(COCCC)=O)C=CC(CNC(=O)Cn2cnnn2)C1 C12(NC(=O)Nc3cccc(OC)c3)CCN(C(=O)COC3CCC3)CC1C2 C1(C2(O)CCOC2)(CC(C(c2ccc(Cl)cc2)NC(C)C=C(Cl)Cl)C)CC1 C=C(C)C(C)(C)C(=O)NCC(C)NC(C1(c2ccccc2OC)CC1)=O c1(C(N2CCCC(N(C(C3CC34CC4)=O)CC)C2)=O)coc2c1CS(=O)(=O)C2 CCC1C(=O)Nc2ccc(C(=O)NCC(C)(CC)NC(=O)C3=CCCS3)cc21 N1(C(C(CCCC)O)=O)C2CCC1C1CC1(NC(C1CCc3nncn3C1)=O)C2 c1(C(N(C2CCN(C(C3(N(C)C)CCCC3)=O)C2)CC)=O)ccc(CF)cc1 c1(C(=O)NC2C(NC(C(CCC)=CCC)=O)CCCCC2)cc2cccnc2s1 CCC(C)C(=O)C(=O)N1CCC2C(C(N3C4CSCC3C4)=O)C2C1 C(C(CNC(C1(C)CCC1)=O)C(F)(F)F)NC(CCc1onc(CSC)n1)=O N1(C(C(C2CCCC2)OC)=O)CC2CCCCC2(CN=c2nn[nH]n2C)C1 c1(C2C(C(=O)NCCCNC(c3cc(F)n[nH]3)=O)C2)cc(F)ccc1F C(CNC1CCCCC1)(CCCC)(c1n(CCOC)nnn1)NCCOC c1(C(N2CC(NC(C=C3CCC(C)C3)=O)C3(C2)CC3)=O)nnn2c1CSCC2 N=c1ccc(C(=O)NCC2CCCCC2NC(=O)CC2(n3cncn3)CC2)c[nH]1 C1(C)(C(N(CC(CN(C(c2nc(COC)sc2)=O)C)O)C)=O)CCC(=O)N(C)C1 N1(C(C2CC(OC)C2)=O)CCCN(C(=O)COc2cccnc2)CC1C N1(C(CSCC(C)C)=O)CC(C)CN(C(=O)CCc2csc(=N)[nH]2)CC1C C1(CC(C)NC(C2CCCCS2)=O)CCN(C(=O)Cc2cncn2C)CC1 CS(=O)(=O)c1ccccc1C(N1CC(CNC(=O)CCC(F)F)C(O)C1)=O C(CN=C(NCc1cccc(OC(C)C)c1)N1CCC(C)C1)N(CC)CC N1(C(c2ccc(C(Cl)Cl)cc2)C(=O)NC(CC)C)CCCC(C)(O)C1 c1(C(=O)NCCN(C(=O)CC2CC2(Cl)Cl)CCC)ccncc1C(F)(F)F Cc1cc(F)c(C(N2CC(NCc3cc[nH]c3)C2)=O)cc1Br N1(C(COCCN(C)C)=O)CCC(CC(N2CC3C=CC3C2)=O)C1(C)C N1(C(Cc2c(C#C)cccc2)=O)CC2CN(C)CC2C1.C12(C)CCCN(C1)C2=O O=C(C1=CC2C=CC1C2)NCC1(C(=O)NCC(O)C2CC2)CCCC1 N1(C(CC=C(C)C)=O)CCC2(CC1)OCCCC2NC(c1ncc(Cl)cc1F)=O C(CN=c1[nH]cnc2cc(C)[nH]c12)(N(C(C(CC)F)=O)C)C1CC1 C1(O)(CCNC(CCC2(C)CCC(=O)N2)=O)CCCN(C(=O)CSCCC#N)C1 N1(C(CCC2C(C)C2)=O)Cc2n[nH]cc2C1C(=O)N(c1cccc(O)c1)C1CC1 N1(C(=O)NC(c2c(OC(C)C)cncc2)C)Cc2cncnc2C(C)C1 Cn1cc(CC(=O)N(CC(N2CC(O)(CC3CC3)C2)=O)CC2CC2)c2ccccc12 C1(C(=O)NCCCC(=O)N2CC=CC2CSc2cccs2)(C(F)F)CC(F)(F)C1 c1(CNC(C(CCC)C(C)C)=O)cnn2c1CN(C(c1c[nH]nc1F)=O)CC2 Cc1c(C(N2CC=CC2CNC(=O)CC2CCSCC2)=O)[nH]c2c(C)cccc12 CC1=C(C(=O)N2CC(N(C)C(C3CC(C)CCO3)=O)C(F)C2)C(=O)OC1(C)C C1(NC(C(c2ccccc2)OC(C)C)=O)CCCC1NC(=O)Cc1cocn1 C1(C(C)C(=O)N(C)CC2CCCN2C(=O)C=CC(=O)NC2CC2)CCCCCC1 Cc1nc(C2CC2)nc(O)c1C(=O)NCCOCCNC(C1CC(C)(F)C1)=O c1(C(N(C2CCN(C(C(CCCC)O)=O)CC2)C)=O)nc(Cl)cc(N)c1Cl c1(C(=O)NCCN(C(C(COC)N(C)C)=O)C)nnn2c1C(=O)NCC2 c1(C(=O)NCCN(C(c2c(C)cc(F)c(Cl)c2)=O)C)cccc2c1CCC2=O CC1COCC(C(=O)N(CC(=O)NC2COCC2O)C2CCC2)O1 c1(CC)nnsc1CNC(=O)CC1CC(NC(=O)CC2OCCC2C)C1 C(=O)(N=c1cc[nH]cc1O)C(c1ccnc(-c2ccc(OC(F)F)cc2)c1)=O.N N1(C(c2cc(F)c[nH]2)=O)CCC(C2CCN(C(c3ccc(F)cc3Br)=O)C2)C1 c1(CC)ccc(C)c(NC(=O)CC2CC(NC(=O)C=CC(=O)N(C)C)C2(C)C)c1 C1(C(=O)NC(C#C)C)C2CCC1CN(C(c1noc(-c3ccccc3)c1C)=O)C2 c1(C(=O)NCCCOCCNC(C2CCC(C)S2)=O)cc([N+](=O)[O-])ccc1N c1(NC(C(C)Sc2nnc(C3CCC3)n2C)=O)nc2ccccc2[nH]1 C(=O)(C(C)(CC)C(N)=O)NC1C(CNC(=O)C=C(C2CC2)C2CC2)CCCC1 c1(-c2c(C)nn(C)c2C)ccc2c(c1C(N1CCCC(C#N)C1)=O)OCO2 C1(C(=O)NC2CC(O)(CNC(C3(C=C)CCC3)=O)C2)CC2CC1CC2O c1(N2CC(NCCO)C2)ncc2scc(Br)c2n1.N1(N(C)C)CCCC(C=O)C1 c1(CC(=O)NC(CC=C)CNC(c2ccn(C3CCC3)n2)=O)ccc(F)cc1Cl c1(C(=O)NC(CNC(C(C=C)(C)CC)=O)(CC)CC)ccc2snnc2c1 N1(C(COC2(C#C)COC2)=O)CCCCCC1CNC(=O)COCCN(C)C CCC(C(=O)N1CC(C)(NC(c2cccc(N3CCCC3)c2)=O)C1)C(C)O c1(SC(C)C(=O)NCC2CC(F)(CNC(=O)C(C)CO)C2)ccccc1 CCCCCC(C)(CC)C(=O)NC1CN(C(=O)CC2CCC(=O)O2)C1 C=C(C)CC(C(=O)NCC(=O)Nc1cnco1)NC(=O)CN(CCCCCC)C C12CN(C(=O)CCCOC)C(CC)(C1)SC(C)C(=O)N2.N1(CC=CC)CCCC1 CC1CN(c2nnc(CN3CSCC3=O)n2Cc2cccs2)CC(C)O1 N1(C(C2(C=C)CC2)=O)CCOC(CCNC(=O)Cc2nocc2CC)C1 CCCCC(O)C(C)C(=O)NOC(CC(C)C)C(=O)N1CC(O)C(O)C1 CON(C)C(=O)CC1(C)CCN(C(=O)CCc2ccc(C)o2)C1 N1(C(c2n(CC#C)ccn2)C(=O)NC(C)(C)CC)CCCN(C)CCC1 c1(OC)ccc(OC(c2n(CC3CCC3)nc(C)c2)=O)cc1I c1(C(N2CC3(CN(C(c4cnc(C)nc4)=O)C3)C2)=O)cnc([N+](=O)[O-])n1C N1(C(c2cc(Cl)c(Cl)s2)C(=O)NCC)CCC(C)(COC)CC1 N1(C(c2nnn(C)n2)=O)CC2CCC(C1)C(NC(C1CC3CC3C1)=O)C2 c1(OC)cnc(CNC(=O)CC(C)(c2ccccc2)C2CC2)c(OC)n1 c1(NC(C2N(C(C(C)(C)CCl)=O)CCC2)=O)cc(Br)cc(C(=O)OC)c1Cl C(=O)(C1=C2CCCN=C2NN1)NC(C12CCC1CN(C(C1CS(=O)(=O)C1)=O)C2)C C1(C(=O)NC2C(C)CCN(C(=O)CSC(C)(C)C)C2)CCOCC12CCC2 CC1CCCCC1(C)n1cc(-c2ccc(N)cc2)nn1.C1(=O)CN1CC1CC1 N1(C(CN(CCOC)C)=O)CCCCC1CC(=O)NCCCC1CCCCC1 C1(N2C(=O)Cn3cc(nn3)C2)CCN(c2ccccc2)CC1.NC(=O)C1CC1 c1(SC)cncc(C(=O)NCC2CC(NC(=O)C(C)C)C2)c1 CCCC(CCC)C(CC)Nc1cc(Br)nn1-c1ncccc1Cl c1(NC(C(C2CC2Cl)OCC)=O)cc([N+](=O)[O-])ccc1C CCC(C(=O)NCC(CNC(=O)C(C)(C)CF)OC)C(C)C c1(C(C(=O)OC2CCCCC2)OC(C(c2ccoc2)SC)=O)cccc(F)c1 C1(C(=O)NC(CCC2CCC2)C(=O)NCC(F)(F)Cl)CC2CCC(C1)O2 N1(C(CC2C(C)CCO2)=O)CCC(CN(C(=O)CC2CCCC2O)C2CC2)CC1 C1(C(=O)NCC(C)NC(c2csc(Cl)n2)=O)CC(=O)CC(=O)N1 c1(C(=O)O)cc(C)c[nH]1.CC#CCCC(C1(C(=O)NCCOC2CC2)CCC1)=O c1(C(N2CC(C)CCC2CC)C(=O)NCCCSCC)ccc2c(ccn2C)c1 C1(C(=O)NC2CC(N(C)C(c3ccsc3)=O)C2)CN2CCN1CC2 c1(OC(C(CC)(CC)CC)=O)ccc2c(c1C(=O)OCC)OC(F)(F)O2 C(CC(CC)CO)NC(C(Cc1cc[nH]n1)NC(CCOCCCOC)=O)=O C1(CCCNC(=O)C=CC2CCC2)CN(C(C2C3CC4C(C3)C24)=O)CCO1 c1(C(=O)NC2C(CCC)CN(C(C3CC3C#N)=O)C2)ncc(C)cc1Br C1(CNC(CC2(C)CC2(F)Cl)=O)CCCCN(C(=O)CC2(O)CCCOC2)C1 C1(CCC)CC(c2nnnn2C2CC(F)(F)C2)(OC)C1.C12CC(C1)CN2 C1(C(N2CCC(C)C(NC(=O)CCCCCF)C2)=O)CC1C1CCCCC1 CC(C)CC(=O)NCC(C(=O)CCO)=O.C(C(F)CNC(=O)C(C)C)N N1(C(c2cccc(CC)n2)=O)CCCC(C)C1CNC(c1cnc(O)cc1O)=O c1(C(=O)NC2C3CN(Cc4c(OCC=C)cccc4)CC32)cc(F)c2cn[nH]c2c1 N1(C(CC(CC)C(C)C)=O)CCCC2(CNC(=O)Cc3ccc(Cl)s3)CCCC12 c1(CC)[nH]nc(Cl)c1C(=O)NCC(C1CCOC1)NC(=O)C=Cc1ccc(C)o1 c1(CO)cc(=NCc2ccc(Cl)cc2NCCl)[nH]c(Cl)n1 C1(COC)CC(CNC(=O)Cc2cnoc2)N(C(c2nocc2C(C)C)=O)C1 Cn1cnc2cc(C(N3CC4(CC(CC(=O)NCC(C)(C)O)C4)C3)=O)ccc12 Cc1cc(C(=O)NC(C2(O)CN(C(C3(F)CCCOC3)=O)C2)C)cn1C N1(C(C(C2CCN(C(C3(C)CC3(C)C)=O)CC2)C)=O)CC(C#N)(CCF)C1 C1(O)(CC(=O)NCCC2(NC(c3scc(C)c3)=O)CC2)COC(C)(C)C1 N1(C(Cn2ncc(C#N)c2)=O)C2CCC1C(CNC(=O)CN1CCCCCC1)C2 c1(C(N2C(C(N(CC#C)CC=C)=O)(CC=C)CCC2)=O)cc(O)nc(O)n1 c1(N(C2CCN(C(CS(CC)=O)=O)C2)CCO)ncnc2sc(C(F)(F)F)nc12 C(c1cccc(Br)c1)=CC(=O)NCCC1CCC(NC(C23CC(CO2)C3)=O)C1 Cc1ccc(C(N2CC3CCC(C2)N3C)C(=O)NC2CCC2)cc1C#N c1(C(N(C)C(c2cn(C)nc2C2CC2)=O)C2CC2)ccccc1O C1(Nc2cn(CCC(=O)N(C)C)nc2)CCC(F)(F)CC1 N1(C(c2c(CC)con2)=O)CCCC1(C)C(=O)NCC1(C)CC(C)C1 Cc1ccc2c(CC(=O)NCC3C(C)CCN3C(=O)Cc3ccsn3)c[nH]c2c1 c12nncn1C2CS.c1(C(C2CC(=C)C2)NCC(F)(F)F)nnnn1CCOC.CC CCCCCCCCC(=O)NC(C)(C)CNC(c1cnn(C2CC2(F)F)c1)=O Cc1ncc(C(N2CC3CC(NC(c4ccc(CSC)cc4)=O)C3C2)=O)c(=N)[nH]1 C1(C2CCOCC2)(C(N2CCC(C)(CNC(c3ccoc3)=O)C2)=O)CCOCC1 c1(C(C)C)c(C(N2CCN(C(c3nnnn3C)C)CC2)=O)nnn1C(C)(C)C c1(C(C(C)C)=O)c[nH]c(C(=O)NC2CN(C(=O)C(F)n3cccn3)C2)c1 c1(C(=O)NCC(C(C)(C)C)NC(CSCCC)=O)cccc(N)c1C C(N=c1ccnc(NCCCn2cc(C(F)F)cn2)[nH]1)C1C(C)(C)CCO1 C1(O)(C(N2CC(C3CCCO3)C2)=O)CCSC1.O=C1CCOCCCN1 C(=O)(CCCCCC(C)C)N(CCCC)C(c1ccc(OC)cc1)C N1(C(C(CC)OC)=O)CCC2CN(C(=O)Cc3cnn(C)c3C)CC2CC1 c1(OC)cc(C(=O)NC(C)COCC(F)(F)F)ccc1CO C(N=c1[nH]c(=NCCCCCCOCC2CC2)[nH]c2c1CSC2)c1c(C)ocn1 C1(NC(C(F)=CC)=O)CC(CNC(C2(N3CCOCC3)CCC2)=O)C(O)C1 Cc1ccc(-c2nc(C3CC(C)(O)C3)n(C3CCOC3)n2)cc1Br C(=O)(C(C)(C)CCCCC)N(C1CC1)CC1N(C(CC(C=C)CCC)=O)CCC1 CCC(O)C(C)C(=O)N1CCC(NC(=O)CC(C2CCC2)C2CCC2)C1C c1(C(N(C2CCN(C(c3onc(C)c3C)=O)C2)CC)=O)ccc(F)c(SC2CC2)c1 C(CCC(=O)N(C(C)C(N1CCCC1CC1CC1)=O)C1CC1)OCCC N1(C(C(CCC=C)(C)C)=O)CCOC2(CCCN(C(=O)CNC(=O)C(C)C)C2)C1 N1(C(C2N(C(C=C(C)C(F)F)=O)CCOC2)=O)CCCC(C2(C)CC2)C1 S(=O)(=O)(c1cccnc1)NC1CCC(C)(CNS(=O)(=O)C2CCCC2)C1 c1(OC)c(C)cc(C(=O)N(CC(C)NC(C2CCCCC(=O)N2)=O)C)cc1Cl O=C(O)C(CCOCc1nnnn1C)Sc1ccc(-c2ccccn2)cc1 C1(O)(C(=O)NC(C2CN(C(c3csc(-c4ccncc4)n3)=O)C2)C)CC(C)(C)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(C)C(NC(c2cc(Cl)cc(F)c2N)=O)CC1 C1(C)(C(=O)NC23CC(CNC(c4cnc(CC)s4)=O)(C2)C3)CCCC1O N1(C(=O)CCc2ccoc2)CCC2(C=C(C(=O)N3CC4CC3C4)C2)C1 C#Cc1ccc(NC(=O)CC2N(C(=O)C(O)CCC(C)C)CCC2(C)C)cc1F N1(C(c2c(C)ccs2)=O)CC(C)(C)OCC1CNC(=O)CCS(C)(=O)=O c1(C(N(C2CCCCC2)CCNC(c2snnc2C2CC2)=O)=O)cc(O)cs1 C1(CC)(NC(=O)C(C)CCOC)CCN(C(=O)Cn2ccnn2)CC1 N1(C(C2(CCC=C)CC2)=O)CC2CS(=O)(=O)CC2(NC(=O)C#CC(C)(C)C)C1 N1(CCNC(N2CC(CS(C)(=O)=O)C2)=O)CCCNC1=O Cc1ccnc(C)c1C(=O)NCC1(C)CCCN(C(c2ccccn2)=O)C1 C1(C(=O)NC2CCC(NC(=O)CN3CCOCC3)C2)CCC12CCOCC2 c1(OCCCC(=O)NCC(CC)NC(=O)C=Cc2cscn2)ccc(CO)cc1 C(c1ccc(F)cc1)=C(C(=O)NCCN(C(CC)=O)CC1CC1)C c1(C(N(CCNC(C2CCCCC2C2CC2)=O)CC)=O)cc2ccc(Cl)cc2[nH]1 CC(CC(=O)NC1CN(C(C2CNC(=O)C2)=O)C1)NC(C1CCCC1)=O c1(C(=O)NCC(=C)CCNC(c2n[nH]c(=N)s2)=O)ccc(C(F)(F)F)c(F)c1 C1(CC(=O)N(C(C)CNC(=O)COCC2(F)CC2)CC)COCC(C)(C)O1 C1(NC(CC=CC)=O)CN(C(=O)CC(O)CN(C)C)CC2(CCC2)C1 C1(C(N2C(C(C)NC(c3cnn(C4CC4)c3Cl)=O)CCC2)=O)CCCC2(CC2)C1 C1(N2CCC(Oc3ccc(Cl)cn3)CC2)Cc2ccccc2O1 N12CCC(CC1)CCNC(=O)C2=O.c1(C(=O)OCC)n[nH]c(CC)n1 C1(NC(=O)OCc2ccc(C)nc2C)CN(C(=O)OC(C)(C)C)CC(C)(C)C1 c1(C(N(CCCNC(C(C)N(C(C)=O)C)=O)CCO)=O)ccn2ccnc2c1 Cc1cccc2c(C(=O)NCC3CN(C(=O)C(C)(C)c4cnn(C)c4)C3)coc12 C12(C(C(=O)NC(CC(=O)OC)C)N)CC3CC(CC(C3)C1)C2 Cn1ncc2ccc(CNC(c3cccnc3-c3ccc(F)nc3)=O)cc12 C(=O)(C1=CCC(F)(F)CC1)NC1CN(C(C2CC(C)C2(C)C)=O)C1 CC1CN(C)CCCN1C(C1CCC1CNC(c1cc2cccn2cn1)=O)=O C1(C(N2CCC(CCOC)(NC(=O)CCC=C(C)C)C2)=O)OCC2CCCCC12 c1(N(C)Cc2ccccc2OCc2c(C)nccn2)cccc2c1CNCC2 c1(C(=O)NCc2cccc(C(=O)NC(COC)C(C)C)n2)ccnc(O)c1F N1(C(c2n[nH]c(C)c2C)=O)CC(NC(c2nn(C)cc2Cl)=O)CC(C)(C)C1 C1(C(=O)NC2C=CCN(C(C(C)c3ccco3)=O)C2)CCCCC12CCC2 C(=O)(C(O)C(F)(F)F)NC1CN(C(c2ccc(COC)s2)=O)C1 C1(C(=O)NC2C(C)CCC2C)C2CCCC2CN1C(=O)C(F)F n1(CC(=O)NCCN(C(C2(C)CCC2)=O)C2CC2)nnc2ccccc2c1=O N1(C(=O)Nc2cc(F)nc(F)c2)CCC12CC1(CCOCC1)C2 C(=O)(C(C)(C)CC(F)(F)F)N1CC(CC)N(C(=O)CCC2CCCCN2C)CC1 Cc1cc2ncnc(N3CCC(NC(=O)C(F)(F)CO)C3C)c2[nH]1 C1(NC(C(C(C)C)OCC)=O)CCC2CN(c3nc(COC)ns3)CC2C1 C1(CC(N2CC(C)(COC)C2)=O)CN(C(c2csnn2)=O)CC12CC2 C1(C(N2CC(C(N3CCC(C)CC3)=O)C(F)C2)=O)CCC(F)(F)CC1 c1(N2C(CCNC(c3ccc(Cl)s3)=O)CCCC2)[nH]cnc2nc(Cl)cc1-2 Cc1ncoc1C(=O)NCC=CCC(=O)NC(C)(C)CC1CC1 c1(C(N2CCC(COC)(NC(=O)C(C)NC=O)C2)=O)ccc2cc(C)ccc2n1 c1(NCc2ccnc(C)n2)c(-c2ccccc2)[nH]c2c(C)cccc12 c1(C(=O)NC(CNC(C(CC)COC)=O)CC)cnn2cc(C(N)=O)cnc12 C(=O)(C1=CC2(CCOCC2)C1)NCC(N1CCCCC1)C c1(OCC)ccc(N)c(C(N2CCC(O)(CNC(=O)CCN3CCCC3)C2)=O)c1 N1(C(CCC2CCC(=O)C2)=O)CCC2CCN(C(=O)Cn3cccn3)CC12 CC1CN(C(=O)COCC2CCCC2)CCC1N(C(=O)CC1(O)CC1)C c1(CNC(C2N(C(C3C(C)CC3)=O)CSC2)=O)cc(F)cc(F)c1 C1(C(N(C(CNC(C2(CCOC)CCC2)=O)C)C)=O)CC=C(C)CC1 C1(C(=O)NCC2CCC(C)N(C(=O)CC3CNC(=O)O3)C2)CCc2nncn2C1 c1(C(c2n(CCOCC)nnn2)NCC2CCCS2)n[nH]c2ccc(C)cc12 CCC1=C(C(=O)N2CCC(NC(c3cscn3)=O)CC2C2CC2)SCCO1 N1(C(C2(CC)CCOC2)=O)CC(CO)C2(C1)CN(C(=O)C(SC)SC)C2 C(=O)(C(F)(F)C(C)(C)O)NCC1CCN(C(c2c(C(=O)OC)[nH]cc2)=O)CC1C CC1(CC(=O)NC2(CNC(c3ccnn3CC#N)=O)CCOC2)CCCO1 C12(NC(C3CNC(=O)O3)=O)CCC(CN(C(c3cccc(C4CC4)n3)=O)C1)C2 c1(C(N2CC(NC(C(=O)NC(C)C)=O)C3C2C3)=O)cc(C#N)ccc1O Cc1nc(C(=O)NCC2CC3CC3N2C(=O)CC(C)C(F)F)c2ccccn12 CC(CF)CC(=O)NCC1(CCNC(C2CC(F)C(=O)N2)=O)CC1 N1(C(C2(C)N(C(C)=O)CCC2)=O)CCC(CO)(NC(=O)C(C)NC(N)=O)CC1 c1(N2CCN(C(C(=O)NC3CC3)=O)CC2)ccc(C(F)(F)F)c(Cl)c1 N1(C(CN(C)Cc2cccs2)=O)CC(F)(F)CC1(C)CNC(C1CNC(=O)C1)=O c1(C(c2n(CCCCCC)nnn2)NCC2CC3CCC2C3)c[nH]c(C)cc1=O c1(OCC#C)cccc(CN2CC(C)(C(=O)NCc3cscn3)C2)c1 C(=O)(CCS(=O)(=O)N1CCCC1)NC(C1CN(C(C2(CO)CC2)=O)CCO1)C c1(C(=O)NCCCCNC(CCOCC)=O)nnn(C(C)(C)C)n1 C1(C2CC2)(CNC(C(CN(C)C)N(C)C)=O)CCN(C(C2(C#N)CC2)=O)C1 C1(NC(CCC2(C)CN(C(c3cc(=N)[nH]cn3)=O)C2)=O)CC12CCOCC2 C1(NC(C(CCC)N(C)C)=O)CC2CN(C(=O)C(C)(C)C3CCCCC3)CC2C1 c1(C(=O)NC(C2OCCN(C(c3c(C)csc3C)=O)C2)C)ncc2[nH]ncc2n1 C12(C(=O)NCCNC(CCCc3ccc(N)cc3)=O)CC=CC(C1)OC2 N(C1CCc2ccc(Br)cc21)C(C(=O)NC(CC=C)Cc1ccccc1)=O C1(OCC(=O)NCCCCNC(C(=Cc2ccco2)C)=O)CCCCC1C N1(C(Cc2cc(=N)[nH]cc2)=O)CCN(C(=O)C2=CCC2)C(C2CCCC2)C1 N1(C(C(CCC)F)=O)CC2CCN(C(C3CCC(=O)NC3)=O)C(C2)C1 C1(CNC(c2cnc(C)o2)=O)CN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC1(C)C C12(C(N3CC(NCc4nc(CC)sc4)OCC3)=O)CCCC1CC(C)CC2 c1(N2CC(CNC(C(C)(C)C(F)F)=O)OCCC2)ncnc2c1CCO2 N1(C(C=C2CCC(C)C2)=O)CCCC(N(C)C(c2cnn(C)c2N)=O)CC1 C1(OC)CCC(C(=O)N(C(C(=O)NCc2c(C)noc2C)C2CC2)C)CC1 C12(CCNC(Cc3c(C)con3)=O)CCC(C1)N(C(=O)CCOCC(C)C)C2 C1(C(=O)NC(C2CSC2)C)(NC(C2CC3CC3C2)=O)CCN(C)C1 c1(OC(CC)C)cc(NC(=O)C(=O)NC(C)(C(=O)O)C2CCCOC2)nc(C)c1 c1(C(=O)NC2CC(CNC(c3cc(C)n(C)c3C)=O)C2)cc(F)c(F)cc1F c1(OC)nc(Cl)ccc1C(=O)NCC(CNC(=O)CC1CCCCC1O)CO N1(C(C=NOC)=O)CC(CNC(C2(Cc3cnn[nH]3)CCC2)=O)C2CC12 c12cc(C)c(o1)C(=O)NC2.c1(COC)n[nH]cc1C(=O)NC1(c2nc[nH]n2)CC1 c1(C(=O)NC23CC(CNC(C=CCN(CC)CC)=O)(C2)C3)cn(C)nc1C C1(CNC(CNS(NC)(=O)=O)=O)CN(C)CCN1C(=O)CSCc1ccnn1C N1(C(C2(C(C)(C)O)CC2)=O)C2CCC(C2)C1C(N1CCCC(O)(C(N)=O)C1)=O N1(CC(=O)NCCN(C(=O)CCCc2cccs2)CCCN(C)C)CCCCC1=O c1(CC)cc(C(=O)NC2(CCNC(=O)CN3CCCCC3C)CC2)c(C)nn1 CCC(O)C(C)C(=O)N(C1CCN(C(c2ncoc2C2CCCCC2)=O)C1)CC C1(CC(=O)N(CC(N2CCCCC2)=O)C)CC2(CCN(CCN3CCNC3=O)C2)C1 C(C(C(=O)N(C)Cc1sccc1C)NC(c1nscc1C)=O)SCC C#CCC(C)(C)C(=O)NCC1CC(n2cc(C(N3CC(=O)NC3=O)(C)C)nn2)C1 C(CCCCC(=O)N1CC2CC2(NC(=O)C=CCCC=C(C)C)C1)NC(C)=O C1(NC(c2ccn(CC)c2C)=O)CCCN(C(=O)C(CC)C(C)C)CC1 C1(C(=O)NCCc2c(C)ocn2)CCC(CNC(C2CC(C)(C)CO2)=O)CC1 c1(-c2scc(NC(c3nnc(CO)s3)=O)n2)cccc(-c2nn[nH]n2)c1 c1(C(=O)NCC(N)C2CC2)noc(C2CCCCC2)c1Br C1(NCc2cnc(C)[nH]2)CCN(C(c2ccc(Br)nc2Br)=O)CC1F C1(C(=O)NCc2scc(CNC(C3(C)CC4CC4C3)=O)n2)C2CC3C(C2=O)C13 CCCC(C)(C)CC(=O)NC1CN(C(=O)Cc2cc(F)ccc2F)CCC1C C1(C(=O)NC(CC)CN(C(=O)Cc2ccccc2Cl)C)CC2C=CC1CCC2 c1(CC)ccc(C(=O)NC2CN(C(=O)CC3(N(C)C)COC3)CC2C)cc1Cl CCC(CC(=O)N1C2CN(C(c3cc(C4CC4)nc(O)c3)=O)CC12)C(C)C C(CC(C)(C)C(=O)NC12CC(C(F)(F)F)(CO1)C2)SC.C12CCCC1CNC2=O C1(NC(CC(COC)C)=O)CC2CCC(C1)N2C(C1(C)CCCO1)=O c1(N(C(C(=O)NCC2CCCO2)C2CCCC2)CC#C)ccccc1 Cc1cc(=O)n(C)nc1C(=O)NC(CNC(=O)CCc1cc(F)ccc1F)CO C1(NC(CC2(C)CCCC2)=O)CN(C(=O)C(F)n2cccn2)C2(CCCC2)C1 CC1CC(NC(c2cccc(C(=O)NCC(F)(F)F)c2)=O)CN1C(=O)C(C)(F)F C12(NC(=O)C=Cc3ccc(Cl)cc3)CCCN(C(=O)CC3CC=CCC3)CC1C2 c1(C(N(C2CCCN(C(=O)COCP(C)(C)=O)C2)CC)=O)cnn2c1CCCC2 C(=O)(CCC(C)CN(C)C)N1CCC(N(CC(C)C)C(c2cnsc2)=O)CC1 c1(CC(=O)NCC(C(C)(C)C)NC(c2cncc(F)c2Cl)=O)c(F)cccc1F c1(CNC2(C(C)NC(=O)CC3CSCCN3)CC2)cnc(Cl)cc1Br c1(C(N(C(CCN(CC)CC)C)C)=O)cncc2c1CCC2.C12(CC1)CC(=O)N2 C(CC(C)N=c1[nH]c(N2CCOC(c3ccco3)C2)nc(=NC)[nH]1)SCC C1(N(C(C(CNC(CC(=O)OCC)=O)N(C)C)=O)C)CCN(C)CC1 N1(C(C(CC)(C)O)=O)CCN(c2cc(-c3ccccc3)ncn2)C(C)C1 c1(C(N(C2CCC(C(=O)NCC(C)(C)C3CC3)C2)C)=O)cnc(N)cn1 N1(CC(=O)NCC(C)CN(C)C(c2nn(C)nc2Br)=O)CCC(O)CC1 N1(C(CC(C)(C)CC2CN(C(c3csc(Cl)c3)=O)C2)=O)CCOC(CO)C1 C1(C2(NC(C=CC=CC)=O)CC2)CCCN1C(c1cnn(CC(C)C)c1)=O C(=O)(CCCCCC(C)C)N1C(CNC(C2CC(C#N)(OC)C2)=O)CCC1 N=c1[nH]ccc(C(=O)NCC2CN(C(=O)CC3CCC3(F)F)CCO2)c1[N+](=O)[O-] Cc1cccn2cc(C(=O)NCCC3CCCN3C(=O)Cn3cnc(=N)[nH]3)cc12 N1(C(C(C)N2CCC2)=O)CCCC12CCN(C(C1CN(C(=O)C3CC3)C1)=O)CC2 C1(C(C(=O)NCCC#N)OC)CCN(C(=O)NCCF)CC1 C1(N(C(=O)CCc2cn(C)cn2)C)CC2CCC(C1)N2C(C1CCCCO1)=O c1(C(=O)NC(CC(C)C)CNC(C2CCC3(CCC3)O2)=O)cnn2ccn(C)c12 O=C(CCC(CF)CF)N1CC2CC2(C(N2CCn3nncc3C2)=O)C1 CCCC(O)C(=O)N(C)CC=CC(=O)NCC1(CCO)CCCC1 CCC(CC)C(=O)N(C)CCNc1nccc(Br)n1 C1(CNC(C=CC(C)(C)N(C2CCCCO2)C(C)=O)=O)(CO)CC2CC2C1 N1(C(c2ccc(CC)s2)=O)CC(NC(C2CN3CCCC2C3)=O)C(C2CC2)C1 C1(C)(CNC(C(N(C(C(CC=CCC)C)=O)C)C2CC2)=O)CCCCCC1 CC1CN(C(=O)C(c2ccccc2)F)CCN(C(C2CC(C)(C)CN2C)=O)C1 C(C(C)(O)CNC(c1ncc(C(F)F)s1)=O)NC(CC)=O C(C)(C(=O)NCC1CCN(C(C2CC(SC)C2)=O)CC1)(C(C)C)OC CN1C(=O)CSC1=CC(=O)N1CC2CCC(CNC(C3(C)CCCCO3)=O)(C2)C1 N1(CC(=O)NC(c2nc(CC)sc2)C)CCN(C(=O)C(C)NC(N)=O)CC1C N1(C(C(CC(C)C)O)=O)CC(NC(C2(F)CCOC2)=O)CCC(O)C1 C1(C(=O)NCC(C)(C)OCCNC(C2C(C)C2)=O)COCCO1 N1(C(C(CSC)OC)=O)CCN(C(=O)Cc2ccc(F)cc2)CC(C)(F)C1 C(=O)(C(C)(C)CC(C)(C)C)NCC1N(C(C(C)CF)=O)CCC1 CCCCC(C(=O)N1CC2(NC)CCC1C2)NC(N)=O.N1CCN(C(=O)C(C)C)CC1 CC(CC(C)(F)F)C(=O)N(C1CCCCC1NC(c1cnn2c1N(C)CC2)=O)C c1(C(=O)NC2C(NC(c3cncn3C3CC3)=O)CC2)[nH]ccc1C1CC1 C1(C(N2C3C(NC(C(c4cccc(Br)c4)C)=O)C(C3)C2)=O)CC12CCCOC2 c1(NC(C)=O)cnccc1C(=O)NC1CC(C(=O)NCc2sccc2C)C(O)C1 N1(C(c2ccc(CCC)cc2)=O)CCCOC(CNC(c2nc(CC)no2)=O)C1 n1(CC)ncc2cc(C(=O)NCC(C)N(C(=O)Cc3ccc(C)s3)C)cnc12 c1(COC)cccc(C(=O)N(C2CCC(NC(=O)C(=O)NC3CC3)C2)C)c1C CC1(C)OCCC1NC(=O)C(c1cccnc1)NC(=O)CC1CC(=O)NC1=O CC(C)CC(C)(CNC(=O)CCCc1ccsc1)NC(c1ccn2c1CCC2)=O c1(C(=O)NCC2(NC(c3c(C)ncs3)=O)CCCCC2)occ2c1CCOC2 Cn1ncc2ccc(NC(C3(F)CCN(Cc4ccc(Br)nc4Br)C3)=O)cc12 CN1CCN(C2CCCN(Cc3cccc(-n4ccnn4)c3)C2)CC1 Cc1cc(C(=O)N(C2CCCN(C(c3cnsc3C)=O)CC2)C)cc(N)c1Cl c1(C(N2CC(NC(CC3N(C)CC=CC3)=O)C2)=O)cc([N+](=O)[O-])c2nsnc2c1 N1(C(CC2N(C(C(CCC)N(C)C)=O)CCC2)=O)CCCC2CCCCC12 Cc1cncc(NC(=O)Cc2ccco2)c1.N12C(=O)CCC1C(=O)O2 c1(N2CCCC(C(C)NC(CS(CC)(=O)=O)=O)C2)cccc(F)c1C#N Cc1cn2c(C(=O)NCC(C)NC(=O)Cc3cnc4n3CCOC4)c(Cl)nc2s1 C(=O)(C#CC(=O)N(C)C)NC1CC(n2cc(-c3cc(C)oc3)nn2)C1 N1(C(c2cnc(C)nc2C)=O)CC2(CCCC2NC(=O)CCN2CCCC2=O)C1 CC(CNC(C1CCCC(=O)N1C)=O)CN=c1[nH]c(Cl)nc2c1CCOC2 C1(C)(C(=O)NC2(C)C(C)OCC2)CCCN(C(=O)C(=O)C2CCCC2)C1 CC1CCN(C(C2(C)CCOC2)=O)CCN1C(c1nc(Cl)sc1Cl)=O CCCC(O)C(CO)NC(c1cnn(CCNC(=O)CC2CC3CCC2O3)c1)=O C1(O)(C(C)NC(=O)Cn2cccc2)CCN(C(=O)C(C2CCCCC2)F)CC1 Cc1ccc(C2CC2C(=O)NCCCCN(C(=O)C(C2CCCCC2)C)C)s1 N1(C(C(C(C)(C)C)NC(c2c(CC)n(C)cc2)=O)=O)Cc2cccc(F)c2C1 C1(CNC(c2n(COC)ncc2)=O)CN(C)CCN1C(C1CCOC(C)(C)C1)=O N1(C(C(C)OCCCCCC)=O)C(C)C2CC1C2NC(c1nn(C)cc1C)=O C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(C2CS(=O)(=O)CCN2)=O)CC1C(N)=O c1(C(=O)NC2C(CNC(CCS(C)(=O)=O)=O)C2)cc(N)c(O)c(F)c1 N1(C(c2c(OCC)scc2)=O)CCOCC2(COCCN2C(c2ccns2)=O)C1 N1(C(C2(Cc3ccccc3)CCN(C)C2=O)=O)CCC2(C1)OCCCO2 Nc1ncnc2c1ncn2CC(=O)OC1CN(c2cc3ccccc3o2)C1 C(C(C)C)(C(O)C(=O)NC(CO)C(C)NC(c1ncn2c1COCC2)=O)OC N1(C(COC)=O)CC2CCC(C1)N(C(c1cc(NC(=O)OC)ccn1)=O)C2 C12(CC(=O)OC)CN(C(=O)C(C)OC)C(CNC(C3CN(C)C(=O)N3)=O)(C1)C2 C1(CC)(CC)CC(NC(c2cc(C)nn2C2CC2)=O)CN1C(=O)CC(C)(C)C c1(C(N2CC3CCN(C(C4C(C)CC4)=O)CC32)=O)ccc(O)c2ccccc12 c1(C(=O)NC2C=CCN(C(C(COC)OC)=O)C2)[nH]c2cc(F)cc(F)c2c1C C(CC(C)C)(C(=O)N(C1CN(C(=O)CC2CCCN(C)C2)C1)C)OC n1(-c2cn(CC)nc2)nc(-c2nc[nH]n2)nc1CCc1cccc(Br)c1 C(=O)(C(CNC(C1CCC(C)(C)OC1)=O)C(C)(C)C)N(C1CCC1)C CCC(CC)(CC(=O)OC)C(=O)NC1CCN(C(=O)C(N2CCCC(C)C2)=O)C1 C=CC1(C(N2CC(C3CCCCC3)C2)=O)CCN(C(=O)CN2CCNC2=O)C1 CC1CN(Cc2ccc(N3CCCC3)nc2)CC1NC(C1CCC1(C)C)=O c1(OC)cnc(C(=O)NC23CC(CNC(=O)CC4CC5(CC5)C4)(C2)C3)c(F)c1 C=C(C)CN=C(NCC1(C(=O)OC(C)(C)C)CC1(F)F)N1CCc2n[nH]cc2C1 N1(C(c2c(SCC)cccc2)=O)CC2CCC(NC(=O)CC3CC3(Cl)Cl)CC2C1 c1(CC(=O)N(C2C3CN(C(C4CCCC(C#N)C4)=O)CC23)C)c(F)cccc1F C=CCC(CC)C(=O)N(CCCNC(C1CC(F)C(=O)N1)=O)C(C)C C12(NC(COCC)=O)COC(C1)C(NC(=O)C(c1ccc(C(F)(F)F)nc1)=O)C2 N1(C(Cc2ccnc(C)n2)=O)CCCC(O)(CNC(=O)C=CC(=O)NC2CC2)C1 c1(C(=O)NCCCn2cc(CCc3ccccc3)nn2)cc(Cl)ccc1Br C12(C=CCN1C(=O)OC(C)(C)C)CC2.C1(COC)CC(O)(C(F)(F)F)C1 c1(C(=O)NC(CC(C)NC(=O)COCCc2cccs2)C)cccc2ncsc12 N1(C(CC2(C)CCN(C(C3C4COCC34)=O)C2)=O)CC2CCC(C1)O2 C=CCCCC(=O)N1CCC(COC)(NC(c2[nH]nnc2C(=O)OC)=O)C1 C1(C2CCN(C(c3cc(C#N)ccc3F)=O)C2)(NC(CCCC)=O)CC1 c1(C(=O)NCC)cccc2c(Br)cccc12.C12CCC(CC1)C(=O)OC2 n1(C(C)C)cnc2c(NC(c3c(F)cccc3F)C)[nH]c(=NCC(F)(F)Br)nc12 C=CCC(C)(CC)C(=O)N1CC(CNC(=O)C(F)(F)c2ccccc2)C(F)(F)C1 C1(CNC(CN(C)C)=O)CCCCN(C(C2(Cc3cccnc3)CC2)=O)C1 C(=O)(CCCCC(C)(C)C)NC(c1ccccc1)C(=O)N(C)CC1(OC)CCC1 c1(C(=O)OC)cc(O)nc(N2CCC(NCc3cccc(Br)n3)CC2)n1 CC(C(C)C(=O)N1CCC(NC(=O)C(C)(O)Cc2ccccc2)CC1)S(C)(=O)=O c1(N(C2CCC(NC(C)=O)CC2)C(c2cc(O)nc(Cl)c2)=O)cccn2nccc12 C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NCCCNC(c1ccc(OC)o1)=O Cc1nc(Cl)[nH]c(=NCC2CCCC2NC(C2(CO)CCC2)=O)c1Cl C(CCCCC(=O)NCC1(O)CCN(C(=O)C(C)C(C)(F)F)C1)=CC C1(NC(C(COC)NC(c2cn(CC)nn2)=O)=O)CCn2nnnc2C1 c1(CC(=O)N(CCN(C(C2C(C(=O)OC)CC2)=O)C)C)cccc(F)c1F C1(NC(C(C)=C2CCC2)=O)CCN(C(C2CN3CCCN2CC3)=O)CCC1CO C12(C(N(CCNC(C(C)(C)N(C)C)=O)C3CC3)=O)CCCC(=O)N1CCC2 CC(C)CC(C)(O)C(=O)NCC(C)CC(=O)NC(CO)C(N)=O C(c1ccncc1)=CC(=O)N(C)CC1(CNC(=O)C=CC(F)F)CC1 c1(C(=O)NCC2CCN(S(=O)(=O)C(F)F)CC2)ccc2c(c1)OC(F)(F)CN2 CCC(CC(=O)N1CCCC1CC(N1CCOC(C2(C)CC2)C1)=O)OC c1(C(C)C)nc(NCCC(F)(F)Cl)cc(=NCC2(C)CCCCC2)[nH]1 c12cnc(c(Cl)n1)CC1CCN2C1.n1(CC)cc(C(=O)NCC(C)=O)nn1 C1(C(=O)NC(c2noc(C)n2)CC)CN(C(=O)CCCCC)CCO1 N1(C(CN(C(C)=O)C)=O)CC(C)C(NC(=O)Cc2ccn(C(F)F)n2)C(C)C1 Cc1cc(C(=O)NCC2CCC(NC(=O)CC3CCCOC3)CC2)cc(C)c1Br c1(OCC)cc(CN2CCCC(CC(=O)NCCC3CCCC3)C2)c(Br)cn1 c1(C(=O)NCCN(C(C2CCNC2=O)=O)CC2CC2)cc(Cl)nc(Cl)c1 N1(C(N2CCCCC(O)C2)=O)C2CCC1(CO)CC2.CC(C)(C)NC(=O)N C12(CC)CC(C(=O)NC3CN(C(c4cnccc4C)=O)CC3F)(CO1)C2 C(C(=O)NC1CC(COC)(NC(=O)COCC(F)(F)F)C1)(C(C)C)SCC c1(C(=O)NC(CC=C)CC(=O)NC(CCCC)C(N)=O)c[nH]c2ccccc12 c1(CC(=O)N(CC(C)N(C(C2CC(CCC)C2)=O)C)C)c(C)nn(C(C)C)c1C N1(C(CC)=O)CCC(C(CC)NC(=O)C(C2CCC2)NC(c2ccn(C)n2)=O)C1 C1(C(NOC(C)(C)C)=O)CC(C)(C)CN1C(=O)COCCc1cccc(F)c1 C(=O)(C#CC1CCC1)NCC1N(C(c2ccc(F)cc2)=O)CCCC1 c1(NC2C(C=C)COC2)cc(S(=O)(=O)NCCC(C(C)C)OCC)ccc1C#N N1(C(C2CC(C)(C)OC2)=O)CCC(NC(=O)C(F)C(F)(F)F)C(F)C1 c1(CNC2C(C(=O)Nc3c(OC)ccc(OC)c3)CCC2)cc(F)c(Br)cc1Cl Cc1cc(O)cc(=O)n1CC(N1CCC(CNC(=O)C(C)C(F)(F)F)C1)=O CCCC(O)C(CO)NC(=O)C(C)(C)NC(=O)CC1CCOC1(C)C c1(C(=O)NC(C2CN(C(CCOCC)=O)C2)C)cccc(N2CCCC2=O)c1 c1(C(N2C(CNC(C3C(C(C)C)OCC3)=O)CC2)=O)cc2c(Cl)cc(F)cc2[nH]1 C1(CNC(C2C(C)(C(F)F)C2)=O)CCC(C(=O)NCCC2CCCO2)CC1 c1(C(N(C2CN(C(CC(CC)SC)=O)C2)C)=O)ccnc2ccnn12 c1(C(=O)NC(C)CCC(=O)NCCn2cnnc2C)coc2c1COC2 c1(C(=O)NCC(CC)NC(C2(CC=C)CCOC2)=O)cc2c(OC)cccc2[nH]1 C1(OC)CCC(CC(=O)N(C(C)CO)C)C1(C)C.C(=O)OC C1(NC(c2cccc(C#C)c2F)=O)CCC2(CCN(C(=O)CC(C)SC)C2)C1 C1(C)(C(=O)NCC2(NC(C=CC(C)C)=O)CCC2)C2CCC(C2)C1(C)C c1(C(N(C2CCN(C(=O)CC3CCCCCO3)C2)CC)=O)sc(CO)nc1C C(=O)(CC1=CCCC1)N1CC(CCC)C(C(=O)NCC(O)C(F)F)C1 C12(NC(=O)C3CC3)CCCC1CN(C(=O)Cc1scnc1-c1ccccc1)C2 C(=O)(C(F)(F)CCn1cccn1)NCC1(NC(C2C(CC)CCCC2)=O)CCC1 N1(C(C(CCC)N(C)C)=O)CCCC(C)(C)C1CNC(c1cccc(OC)c1C)=O C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)C(c2ccnn2C)O)CC1)N(C)C CCC(C(=O)N1CC(C(=O)Nc2ccc3[nH]ncc3c2)(SC)C1)C(F)(F)F C(=O)(C1=CCCOCC1)NC1C(C(N2C(CC)CC(C)C2)=O)C2CCC1C2 C(C(C(F)(F)F)N1CCOCC1)NCC(=O)NCC(=O)NC1CC1 C1(COC)CCC(C(N2CCCC2CN(C(=O)Cc2cc(C)ns2)C)=O)C1 C12(CNC(=O)CC3CSCCS3)CCC(C1)N(C(c1cc(O)cc(F)c1)=O)C2 N1(C(C2N(C)CCC2)=O)CC=C(CNC(=O)Cc2cnsc2)CC1 c1(OC)ccc(C(=O)NCC(C2CCCC2)NC(=O)CC(C)F)c(OC(C)C)c1 C(=O)(CC(C)(C)NC(c1ccn(CC)n1)=O)NCc1cnc(CC)[nH]1 CCC(CC(F)(F)F)C(=O)NC(CN(C)C(c1ccc(NC(N)=O)cc1)=O)CC c1(C(N2C3(C(N4C(C)CC5(CC5)C4)=O)CC3CC2)=O)ncc2ccccn12 C(C1=NOC2CN(C(=O)CCn3nc(C)cc3C)CC12)NC(C=CCCC)=O C1(CNC(C(C)(Cl)Cl)=O)CC2CC2N1C(c1cc(Br)ccn1)=O C(N=c1[nH]c(=NC(C)CC)[nH]c2cccnc12)c1ncc(CC)nc1 N12CCC3(C1)CN(CCO3)C(=O)c1cncc(c1)C2=O.C1(OC)CC(C)N(C)C1 CC1CN(Cc2cn[nH]c2)CC1NC(=O)NC1CC12CCCC2 C1(C(=O)NCCN(CCOC)C(c2cc(F)c[nH]2)=O)CC(=O)NC(C)C1 C(=O)(C(O)C(C(C)C)OC)NC(C(=O)N(CCC1CC1)CC)CCSC C1(C(=O)NC2CC(NC(C34CCC(CC3)OC4)=O)CC2O)CCC2(CCC2)O1 C(CN=c1[nH]cc2ncnc-2[nH]1)C1CCN(C(=O)CC2CCS(=O)(=O)C2)CC1 N1(C(c2cn(C)nc2)C(=O)NC2CC2)CCCC2(C=CCO2)CC1 c1(C(N(CC(CNC(c2scc(C)c2)=O)C)C)=O)cc2ccncc2[nH]1 c1(CC(C(=O)NCC(C(C)C)NC(C2CC3(CCC3)C2)=O)C)cccc(F)c1 N1(C(c2cc(C(C)C)nn2C)=O)CCCN(C(C2CCCC(=O)N2)=O)C(CO)C1 C1(CNCC(=O)Nc2ccc(OC)c(OC(C)=O)c2)CCc2ncn(C)c2C1 N1(C(C(C(C)(F)F)F)=O)Cc2c[nH]c(=N)nc2C1 Cc1nc(C(C)C)nc(C)c1C(=O)NCC(C)CNC(c1nc(C2CC2)cs1)=O c1(NC(c2ccc(CCC)s2)=O)cccc(NC(C2CCCSC2)=O)c1 C12(C(N(CC(C)(C)O)C)=O)CCC(CN(C(=O)CC3CCSCC3)C1)C2 C1(CC(=O)OC)CC2(CC2)CN1C(C)=O.c12cc(ccc1I)NC(=S)N2 C1(NC(c2nc(CC)sc2N)=O)CC2CN(C(c3ccc(NC=O)cc3)=O)CC12 N1(C(C(CCC)O)=O)CCCC(O)(CNC(c2ccc(C(=O)NC(C)C)cc2)=O)C1 Cc1nc(C)c(C(=O)NC(CNC(c2cn(CC(N)=O)nn2)=O)CO)c(C)n1 C1(C(=O)NC(C2CCN(C(CSCCOC)=O)CC2)(C)C)CCc2cnnn2C1 Cc1cc(NC(c2ccc(O)nn2)=O)ccc1NC(c1n[nH]c(C)c1F)=O c1(OC)n[nH]c(C(=O)N(CC(C)N(C(=O)C(c2cccnc2)O)C)C)c1Cl N1(C(CCSC)=O)CCC(C(=O)NC2CCN(C)CC2)C(c2ccccc2)C1 C1(CNC(C2C(OCC)C2)=O)CCN(C(c2nnn(C)c2C(F)F)=O)CC1(F)F CCC(C(=O)N(C1CCN(C(c2csc(C)c2)=O)C1)C)C(C)(F)F CC(C)CC(C)C(=O)N(CCCCN(C)C(C1(c2cccnc2)CC1)=O)C N1(CC)CCC(C(=O)NC2CC(OCC(=O)NCC3(CC)CCCC3O)C2)CC1 N1(C(CNS(C)(=O)=O)=O)CCOC(CNC(c2cccc(CC(F)(F)F)c2)=O)C1 C1(CNC(C2CC(OC)C2)=O)CCN(C(C2CCCCCC2)=O)CC1 c1(CC)cc(C(=O)NC2CCCC(NC(c3cncnc3C)=O)C2)cn(C)c1=O C(=O)(CCN(OC)C(=O)c1c(C)cccc1F)Nc1ccc(CC)cn1 CC1(C)CN(C(C2CCC(O)CN2C(=O)CSCC(N)=O)=O)CCCO1 C1(NC(C2CC(=C)C2)=O)CCN(C(=O)C=Cc2ccc(C)c(C)c2)C12CCCC2 c1(C(N(CC(C)(C)NC(C2CCC(C)(C)O2)=O)C)=O)cc(Cl)cc(Cl)c1F N1(C(=O)CC2CC3CCC2O3)CCC2CN(C(=O)C(F)(F)C3CC3)CC2C1 c1cccc2c1CC(C)(C)O2.C(C(C)(C)O)OC(=O)OCC.C1(=O)CN1CCOC N1(C(C2CCC(CC)O2)=O)CC(O)CC1C(N1CCC(COC)CC1)=O C1(NC(C2N(CC)CC2)=O)(CO)CN(C(c2cc(C3CC3)no2)=O)C1 C1(C)(CNC(C2(OC(C)(C)C)CCCC2)=O)CCCOC1.N CCCCC(O)CCC(=O)NCCC1CCN(C(=O)C(c2cccc(O)c2)C)C1 c1(CC)cc(C)ccc1C(=O)NCC1(COC)CCCN1C(C1CCC1(F)F)=O C1(NC(c2ccc(F)cc2)=O)CCCCCN(C(C2CC3CC2C3)=O)C1 C1(CC(=O)NC(C=C)COC)CCCN(C(=O)C(=O)NOC)CC1 c1(C(N(CCN(C(C)C)C(C2C3COCC23)=O)C)=O)ccc(S(=O)(=O)CF)nc1 c1(C(c2cccc3nc(C)sc23)C2CN(C(=O)NC)C2)ccc([N+](=O)[O-])cc1F c1(CC)ccc(C(N2CC(NC(=O)C3CC3)C3CC23)=O)nc1 c1(CC(=O)NC(CNC(c2c(C)occ2)=O)(C)C)cc(C(F)(F)F)nn1C N1(C(CS(=O)(=O)NC(C)(C)C)=O)CC2CS(=O)(=O)CC2(C(=O)OC)C1.C(=O)CO Cc1cc(C=CC(=O)NCC2COCC2NC(C2CC(=O)N(C)C2)=O)on1 C(=O)(CCC(=O)NC1CC1)NC(C=CC(N1CC(C2C(CC)C2)C1)=O)C c1(CN2CC(NC(c3ccc(Br)cc3)=O)CC(F)(F)C2)cn2c(Br)cccc2n1 c1(NCC2(NC(c3[nH]nc(OC)c3Cl)=O)CCCC2)nc2c(cc1Cl)C(=O)OC2 C1(C(=O)NCC2N(c3ncc(C(=O)OC)cn3)CCC2)CCC=CCCC1 c1(OCCCC)ccc(C=NOCC(=O)Nc2ccc([N+](=O)[O-])cc2)cc1 C(=O)(CCCCCC(C)C)NCCCCC1CN(C(c2cc(C)cc(F)c2)=O)C1 C(=O)(CC(C)NC(=O)C(c1ccn(C)c1)C)NCC1CC(=C)C1 C(=O)(C1=NOCC1)N(C1CCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1)C C1(COC)CN(C(=O)C=CC(C)NC(=O)Cn2cc(Cl)cn2)C1(C)C C(=O)(C1=NOC(CN)C1)NCC1(F)CC(NCCC2(C)CC2)C1 N1(C(C2SCCN(C(c3ccc(C(F)(F)F)nc3)=O)C2)=O)CC2CCCC2C1 C1(O)(CC(=O)OC)CCN(C(c2cccc(-n3nnnc3O)c2)=O)C1 C12(NC(C(F)=CC)=O)CCC(CN(C(c3cnc(OCC)cn3)=O)C1)C2 c1(N2C(=O)CC(C(N(CCCNC(C(CC)SC)=O)C)=O)C2)c(C)nn(C)c1C N1(C(c2c(C)cc(C)c(C)c2)C(=O)NCC(F)F)CCC2(CC1)CN(C)C(=O)O2 O(NC(=O)C(CNC(=O)C=NOC)N(C)C)CC#C C1(NC(COC)=O)CN(C(=O)Cc2c[nH]nc2C)C2(CCC2)C1 N1(C(C(CC)OCC)=O)CC=C(C(=O)NC2(C)CC2(C)C)C1 C12(CC)CN(C(=O)COC)C(CNC(c3ccc(C(N)=O)[nH]3)=O)(C1)C2 C(=O)(C1=NOC(C)C1C)Nc1c(C)cc(NC(=O)CCc2nc[nH]n2)cc1 C1(C)(C(N(CC(C)(C)NC(CCCC(=O)OC)=O)C)=O)CCC(F)(F)CC1 Cc1c(CO)cccc1C(N1CCOC(C(C)(C)C)C1)C(=O)NCCSC c1(CSCCNC(C2C(C(=O)OC)C2)=O)ccc(C)c(F)c1.c12cn-1nn2 c1(C(=O)NCC2CCC(NC(C(C)SCC)=O)CC2)nccc2ccncc12 c1(C(=O)NC2C(CNC(=O)CCSC3CCCO3)C2)ccc2cncn2c1 c1(C(C)C)n[nH]cc1C(N1CCCC1C(=O)NCC(C)N(C)C)=O C12(C(N(C(c3ncccn3)C)C)=O)COCC1CN(C(=O)Cc1ccccc1)C2 C1(CNCc2cc(OCCCOC)c(OC)cc2)CCc2ccccc2C1 C=CC(C)(O)C(=O)NC1CC1NC(c1cc(Br)ccn1)=O Cc1cc(Cl)c(C(N2CCCCC2CC2CCCC2)=O)s1 N1(C(=O)CCn2cncn2)CCCC2(C1)CN(C(c1cnsn1)=O)C2 N1(C(CN(C(C(F)(F)F)c2cnn(C)c2)C)=O)CCCc2ccc(NC)cc21 c1(CONC(=O)C2CCC2C)ccccc1C1(Cc2cn(CC)nn2)CC1 C(=O)(C1CCc2ccc(Cl)nc21)NC1CC(NC(C(C(=O)OC)C)=O)C1 C1(NC(C2(NC(Cc3nn(C)c(CO)c3)=O)CC(O)C2)=O)CCC=CCCC1 c1(C(=O)NC2CCC(NC(c3cc(COC)on3)=O)C2)cccc(Cl)c1C c1(C(=O)NCC2CC(C(F)(F)F)(CNC(c3c(OC)scc3)=O)C2)nnn(C)c1N CCCCCS(=O)(=O)CC(=O)N(C)CCOCCN(C)C(c1c[nH]c(C#N)c1)=O CC(C)CC(CNC(C1CCOC1(C)C)=O)C(=O)NCc1ncc(CO)[nH]1 C(=O)(C1(CC)CCC(=O)c2ccccc21)NC12CC(NC(C(F)=C(C)C)=O)(C1)C2 c1(COC)cc[nH]c1C(=O)NCC1CC1CC(=O)NCCC1CCC2CC12 n1(C(CC)C)ncc(C(N2CCC(NC(C3CC(=O)C3)=O)C2C)=O)c1C C(C(C)C)(C(O)C(=O)N1CCN(C(c2cn(C)nn2)C(=O)NC(N)=O)CC1)OC c1(C(N2CCC(CN(c3ncc([N+](=O)[O-])cn3)C)C2)=O)c[nH]nc1S(N)(=O)=O n1(CCC(=O)NCC(C)(C(C)C)NC(CNC(C)=O)=O)cc(C#N)c(O)nc1=O c1(CC)cc(NC(=O)C(C2CCC2)NC(=O)C(CCOC)OC)ccc1C N1(CC(=O)NC2C=CCN(C(C=CCC)=O)C2)C(=O)c2ccccc2S1(=O)=O c1(C(N2CCC(CNC(C(C)n3ccnn3)=O)CC2)=O)nnn2c1C(=O)NCC2 CC(C)(C#N)CC(=O)c1n2c(nn1)CC2.C1(C(F)(F)F)(NC2CCOC2)CCCC1 c1(NC(C2(C)CCN(C(C(C)NC(C)=O)=O)CC2)=O)ccc2nsnc2c1 CCC(C#N)(CC)C(=O)N1CCC(C(=O)NCC2(O)CCCCC2)CC1 c1(C(N(C)CCOCCCN(C(=O)C(F)n2ccnc2)C)=O)ccc2c(c1)CC2 C1(C)(C(=O)NC(C2CCN(C(=O)Cn3cc(Cl)cn3)C2)C)CC=CC1 Cc1ccc(O)c(CC(=O)NCCC2CN(C(c3n[nH]c(C)c3Br)=O)C2)c1 C1(n2cc(CC(C)C)nn2)CCCC(C(=O)O)C1.C12CN(C1)C(=O)CO2 c1(-c2ccc(NCC(c3ccccn3)O)o2)cccc2cccnc12 N1(C(C2N(C(CC)=O)CSC2)=O)C2CCC1(CNC(=O)Cn1cncn1)CC2 C12(CC)CC(NC(=O)CC3CN(C(=O)C(C)CCOC)CCO3)(CO1)C2 N1(C(c2cc(C)c(C)[nH]2)=O)CCCCC2(CCN(C(=O)COCP(C)(C)=O)C2)C1 CC(C)C1=CCC(C(N2CCC(CN(C(=O)CCCS(C)(=O)=O)C)CC2)=O)CC1 c1(CC(=O)NCC(C(C)C)(C)NC(=O)Cc2sc(O)nc2O)ccc(Cl)c(F)c1 CC(C)C(O)CC(=O)NC(C1CN(C(=O)C(c2ccc(F)cc2F)(F)F)C1)C c1(NC(CN2CCN(Cc3c(OC)ccc(Br)c3)CC2)=O)ccc2nc(C)oc2c1 C=CCC(CC(=O)N=c1cc(OC)n(C)[nH]1)NC(=O)CCCNC(C)=O C1(NC(c2c(CC)scc2)=O)CCN(C(C2COCCN2C(C)=O)=O)CC1(C)C c1(C(=O)NC2CC3(C(NC(c4cc(C(C)=O)sc4)=O)C3)C2)cc(C#N)ccc1N C1(C2CCN(C(=O)C3=NOC(C)C3)CC2)(NC(CCCCOC(C)C)=O)CCC1 c1(NC)cccc(C(N2CCCCC2C2CCN(C(C3CCOC3)=O)CC2)=O)n1 c1(CC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)CN2CCC(C)C2)cn1 Cc1nn[nH]c1C(N1CC(N(C)C(C2CCCC2C)=O)C1)=O CC1CC(NC(C2CN(C(c3ccccc3)=O)CC2C)=O)C(=O)O1 N1(CC)C2CCC1CN(C(=O)CCCCN(C(=O)CC1CCCO1)C)C2 c12ccc(c(F)c1)S(=O)(=O)NC13CCC(CC1)(C(N(C)C)C3)C(=O)O2.CCSC N1(C(c2c(CNC(C(CC=C)(C)O)=O)nnn2C)=O)CCC2CCN(C)CC12 C1(N(C(Cc2nc(CC)sc2)=O)C)CCN(C(c2cn(C)c(C)n2)=O)CC12CC2 Cc1c(O)nc2ccccc2c1C(=O)NC1CC1NC(=O)C(CN(C)C)C(C)C C1(N(C(=O)C(c2nc(C)cs2)C)CC)CCCN(C(=O)CC2CCCCC2C)C1 C1(n2c(-c3c(-c4nccc(SC)c4)cc(C)cc3)ncc2)CC12CCN(CC#N)CC2 C=C=CC(C)C(=O)OC(C1CCN(C(c2ccc(OCC)nc2)=O)C1)C N1(CC(=O)NCC2N(C(C(COCC)(C)C)=O)CCCC2)CC(=O)N(C)C1=O N1(C(c2c(OC)scc2)=O)CC(NC(=O)C(C(C)O)NC(C)=O)CC(F)C1 C1(O)(CNC(C(C)=CC)=O)CC2CCC(C1)N2C(c1cc(CC)n(CCO)n1)=O c1(C(N2CCN(C(CNC(C(CCSC)O)=O)C)CC2)=O)nccc(C)c1F S(=O)(=O)(c1c[nH]c2c(Cl)cccc12)NC1CC(CC(=O)O)C12CCC2 C(=O)(C1Cc2c(Cl)cccc21)NC1C(NC(CC(=O)OCC)=O)CC1 N1(C(C2C(C)CCS2)=O)CCC(C)(C)C(CNC(c2cc([N+](=O)[O-])cn2C)=O)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCCC(N(C)C(c2cc[nH]n2)=O)CC1 CN1C(=O)NCC1C(=O)NCCC1CN(C(=O)CCSCc2ccccn2)C1 C(=O)(CCCC(C)(C)C#N)NC1CC(N(C(=O)CC(C=C)C)CC(C)O)C1 N1(C(c2cc(C)sn2)=O)CCCC2(NC(=O)CCC3CCC(=O)N3)CCCC12 C(=O)(C(CCC1CCC1)SC)NCC(CNC(C12CCCC1C2)=O)OC Cc1cnc(SC(CN(C(=O)C(N2CC(F)(c3ccn(C)n3)C2)=O)C)C)o1 N1(C(C(CC(F)F)N(C(=O)Cc2ccsn2)C)=O)CCOCC(F)(F)C1 C12(C(=O)NCCN(CCC)C(c3cncs3)=O)CC(C)(C1)OC2C C1(CNC(c2nn(C)c(O)c2)=O)CCN(C(c2ccc(C(C)(C)C)[nH]2)=O)C12CC2 C1(c2n(CCCOC)nnn2)(Nc2ccc(C)nc2OC)COCCC1C C12(CNC(c3sccc3C(F)F)=O)CC(CN1C(=O)C=CI)C2 c1(C(=O)NC2CCC(NC(c3ccc(SC)cc3)=O)C2)cc(SC)cc(Cl)c1 CC(C)CC(CC(C)C)C(=O)NC(C)CC1CN(C(C2CS(=O)(=O)C2)=O)C1 N1(C(CC(CC)O)=O)CCC2(CCCC2NC(=O)C(C)(O)c2ccccn2)CC1 C1(NC(C(N2CCOCC2)C)=O)CC2(C1)CC2NC(=O)C(O)Cn1cncn1 c1(CC(=O)NC(CNC(c2nnn(C)c2N)=O)C2CC2)ccc(Cl)cc1[N+](=O)[O-] N1(C(CC=C)=O)CCC(NC(C2(Cc3cccnc3)CCC2)=O)CC1 CCCCC(C(=O)NCc1ccnc(C(=O)NCCC(=O)NC)c1)N(C)C Cc1nccc(CCC(N2CCC(C(C)NC(c3coc(C)n3)=O)CC2)=O)n1 C=C(C)CCCC(=O)N1CCC1.c12c[nH]c(c1)C(=O)N(C)C(=O)C2 Cn1ccn2ncc(C(N3CCC3C(=O)N(CC(C)(C)C)CCO)=O)c12 c1(C(N(CC(C)N(C)C(c2cscc2Br)=O)C)=O)ccc2cc[nH]c2n1 C(C)(C)(C(=O)NCC1(O)CC(CNC(c2cnc(N3CCOC3=O)s2)=O)C1)SC Cn1nc(Br)cc1CC(=O)NC(CNC(=O)CNC(=O)NC1CC1)C1CCC1 c1(-n2ncc(C(N(C)CCN(C)C(C3CCC(C)(C)O3)=O)=O)n2)ccc(Cl)cc1 C1(CC2CCC(C(N(C)C)=O)O2)CC2CCC1O2 C1(C(N2CC(O)(CNC(CCC=CC)=O)C2)=O)Cc2ccc(F)cc2O1 CC(C)CC(F)C(=O)NCC(C)CN(C(=O)CNc1nccs1)C N1(C(c2cnc(SC)nc2O)=O)CCC2C(C1)CN2C(c1c(C)cccc1C)=O C1(CNC(C(CC#C)C2CC2)=O)COCCN(C(c2cc(C)n(C)c2)=O)C1 CC1CCC(=CC(=O)NC(C2CCCN(c3nc(CC4CC4)ns3)C2)C)CC1 C(=O)(C(CC1CCCC1)NC(c1nnsc1N)=O)N(C)CCO N1(C(C(C2CN(C(=O)C(C(C)C)SC)C2)OC)=O)CC2CCCC2C1 C12(CNC(C(CC)CC)=O)CCC1CCN2C(=O)C(c1c(C)noc1C)C N1(C(C=C(C)Cl)=O)CCN(C(=O)Cc2ccnc(F)c2F)C(C(C)C)C1 c1(CC(N2C(C3(O)CN(C(C(CC)SC)=O)C3)CCC2)=O)cc(Cl)ccc1Cl n1(CC)c(C)cc(C(=O)NC(C2CCOC2)CNC(c2cn(C)nn2)=O)c1C Cc1ccc(C(=O)NC23CC(CNC(c4csc(O)n4)=O)(C2)OC3C)c(F)c1 C1(C(=O)NCC(CC)(C)O)CC1C1CN(C(=O)CC(Cl)Cl)C1 c1(C(=O)NC2CCN(C(CCCN(C)C)=O)CC2O)cc2cc[nH]c(=O)c2s1 c1(C(=O)NC(CNC(C(c2cccc(N)c2)O)=O)CO)cnc2n1CCS2 c12ccc(cc1)CN(C)CC(=O)N2.c1(CCC)sccc1C(=O)OC c1(N2CCC(C(N(C)C)=O)CC2)nc(Cl)nn2cccc12 C=CCC(C(=O)NCC1(C(N)=O)CN(C(c2cnc(S)n2C)=O)C1)NC(C)=O C(=O)(C1=NNC(=O)CC1)C(C)(C)CNC(=O)CNC(c1ncccn1)=O N1(C(c2c(C)snc2)=O)CCC(NC(=O)C2=NOCC2)C(C)C1 C(=O)(C1=CCSC1)NC1(CCNC(CC=C)=O)CC1c1ccccc1 C#Cc1cc(NC(C2(C)CN(C(=O)CC(C)CC)C(C)(C)C2)=O)ccc1C N1(C(C(=Cc2ccncc2)C)=O)CC(CNC(c2csc(Cl)n2)=O)OC(C)(C)C1 c1(OCC(=O)NC(COC)Cc2ccccc2)ccc([N+](=O)[O-])cc1F C(=O)(C(C)(CNC(=O)C(C(=O)NCC)C(C)C)S(C)(=O)=O)OCC.C(C)(C)(C)OC=O C1(C(=O)NCC2(CCNC(C=C(C)C)=O)CC2)CC2CC(C1)CC(F)(F)C2 C1(CCNC(CCOCCN(C(C2(N(C)C)CCC2)=O)C)=O)CCCC12CC2 C#CC1(O)CCN(C(=O)CC(COC)NC(=O)CNC(=O)C(C)CC)C1 c1(C(N2CC(O)(C(CNC(C(CN(C)C)O)=O)(C)C)C2)=O)cc(N)ccc1Cl C(=O)(CCN(OC)C(=O)C(CNC(C1(C)CC(=O)C1)=O)OC)OC C(=O)(C(C(C)(C)C)NC(N)=O)NCC(CNC(Cc1n(C)ncc1)=O)CO N1(C(c2cnc(CC)s2)=O)CCC(CNC(=O)CC(C)C2CCCC2)CC1 N1(C(Cn2c(C)ccc2C)=O)CCC(NC(=O)COc2cccnc2)CC1C C1(C(=O)NCC2CN(C(CC3CC(SC)C3)=O)CC2C)CCc2nnn(C)c2C1 C(=O)(C(C)(O)CC(F)F)NCc1c(CN(C(=O)CCCF)C)cccc1 N1(C(C2N(C(C)(C)C)CC2)=O)CC(NC(c2ccc(Br)c(Cl)c2)=O)C(C)(C)C1 C1(C(=O)OC)CN(c2ccccc2)CCN1C(=O)CCOc1cccc(Br)c1 N1(C(c2ccc(N(C)C)s2)=O)CC2CC(N3CCCCC3CCO)C1C2 C(CC(F)(F)F)(c1ccccc1)NCC(c1noc(-c2cccs2)n1)=O N1(C(c2c(SC)n(C)nc2)=O)CCN(C(C2CCS(=O)CC2)=O)C2CCCCC12 c1(N(C(c2cc(CC3CCN(C(C)=O)CC3)no2)=O)C)ccc([N+](=O)[O-])c(C)c1 CCCC(C(=O)NCC(C)(O)CO)NC(=O)C=Cc1ccsc1 C1(NC(C23N(C(c4cc(C(C)C)no4)=O)C(CC2)CC3)=O)CC(O)CC(C)(C)C1 C1(OC)CN(C(C2OC3CCC2C3)=O)C(C)(CNC(C2CC(C)(C)CCO2)=O)C1 c12ccc(c(C)n1)c1ccc(cc1F)c(=O)[nH]2.c1(SCCCC)nc[nH]n1 c1(C(=O)NCCCC(C)NC(C2CCSC2)=O)ccccc1F Cc1cn2c(CCC(N3CCN(C(c4scnc4Cl)=O)C4CC34)=O)csc2n1 c1(C(N(C2CCN(C(C3CNC(=O)C3)=O)C2)CCC)=O)coc2c1CCCC2 N1(C(C(c2n(C)ccc2)=O)=O)CC2CC1CN2S(=O)(=O)Cc1ccc(F)cc1F C1(C(=O)NCC#CCNC(Cn2c(C)cc(C(F)F)n2)=O)CCCC(=O)N1C C1(NC(c2c(CC)oc(C)c2)=O)CN(C(C2CC(=O)N(C3CC3)C2)=O)CCC1F c1(N2CC(NC(CCC#CC)=O)C(C)CC2)nc(C(C)(C)C)ccc1C#N c1(N2CCCC(C)(COC)C2)nc(=NCCC2CC(C)(C)CO2)[nH]c2c1COC2 NS(=O)(=O)CCCNC(C1CC=CCC1NC(c1ccc(CC#N)cc1)=O)=O C1(CCCNC(C(C)(F)F)=O)CCN(C(c2cc(Cl)no2)=O)CC1 c1(OCC(C)C)ccc(CSCC(=O)NC2COC(C)(C)C2)cc1 CN=S(C)(=O)CCNC(=O)NC1C=CCCC1C C1(S(N)(=O)=O)(C(=O)NC2CN(C(c3cn(-c4ccc(C)cc4)nn3)=O)C2)CCC1 C(=O)(CCCS(N)(=O)=O)NCC1CCC(F)(CNC(c2cn(C)nc2)=O)C1 Cc1nnc2n1CCC(C(=O)OC(=O)C1CC1)C2.N1S(=O)(=O)NCC1 C1(C#N)(C(N(CCCC(=O)NCCC2ON=C(C)C2)C)=O)CC1(C)C CN1CC(C(=O)NCC2CC2NC(=O)Cc2nn(C)cc2Cl)CC1=O C(=O)(C(=O)NNC(=O)C1CC1c1ccc(C2C(C)(C)C2)cc1)ON1CCC(N)CC1 C1(NC(C2C3(CCN(C(C4(C#N)CC4)=O)CC3)C2)=O)CCOC2(CCOCC2)C1 C(c1c(Cl)nc2ccccn12)=CC(=O)NCCOCCCN(C(C=CSC)=O)C C=CCC(CC(C)C)C(=O)Nc1cccnc1CNC(=O)C=Cc1ccco1 C1(CNC(CC)=O)CCC2(CC1)CCN(C(C1(COC)CCCO1)=O)CC2 c1(C(=O)NCC(C)(C)NC(C(CCC)NC(N)=O)=O)cnc2n1CC(C)CC2 c1(C(N2CCC(C(=O)NCCCOC)(OC)C2)=O)cnc(O)cc1C C1(CC#C)CCCCN1C(c1csc(CNC(=O)C(c2ccccc2)O)c1)=O C1(CCN(C(=O)C(C#N)C2CC2)C)CCCCN1C(c1cncs1)=O c1(C(=O)NC2CN(C(c3occc3Cl)=O)CC2)c(Cl)ccc2ccncc12 c1(CNC(C23CC(C2)C3)=O)nc(C(=O)NCCC2CC2)cs1 C(CC)(C(=O)NCCN(C(C)CC)CCOC)NC(COCCC)=O C1(CCNC(c2c(CC)nns2)=O)CCCN(C(=O)CS(=O)CC)CC1 c1(C(N2C(CNC(Cn3ncc(C)c3)=O)CC2)=O)c(C)ccc(C)c1C C(C(C)(C)C1=CCCC1)SCC(c1n(CC(=C)C)nnn1)(C)NC(C)C1CC1 c1(N2CCCC(CNC(c3ccc(O)nn3)=O)CC2)nc2ccc(O)cc2s1 C(=O)(C(F)C(C)(C)O)N(C)Cc1cccc(CNC(C(C)(C)OC)=O)c1 CC1(C)CCN(C(c2cccc(N)c2)=O)CC1NC(=O)C=CCF N1(CCC(=O)NC2(C)CC(NC(c3cn(CC(C)C)nc3)=O)C2)CCC(O)CC1 Cc1cnc(N)c(C(=O)NC2CC3(C2)CC(NC(c2cc(Cl)ccc2F)=O)C3)c1 c1(C(C)C)ccc(C(N2CC3CC2(c2cn(C4CCS(=O)(=O)C4)nn2)C3)=O)cc1 c1(C(=O)NCC2(F)CCN(C(CCC(C)OC)=O)C2)c(C)c(C)cc(C)c1C N1(C2CC(C(=O)NCC(CCOC)NC(C3COCCO3)=O)C2)CCN(C)CC1 c1(N2CC(C)C(C)C2)nc(N(C)CC2(C#N)CC2)c2ncn(C)c2n1 c1(OC)nc(C(N2CCCC2CNC(C2(OC)CCC23CCC3)=O)=O)cc(O)n1 C1(CN(C(=O)CCC2CCCC2)C)CCN(C(c2c[nH]nc2C2CCC2)=O)C1 c1(C(N(C2CCCN(C(=O)Cc3ccc(Cl)cc3)C2)CC)=O)cncc(CO)c1 C#Cc1ccc(C2(C(=O)NC3C4CCC3N(C(=O)Cc3ccsc3)C4)CC2)cc1 CN1CCCCC1C(=O)NC1CC(CCN(C(=O)CC2CC(F)(F)C2)CCO)C1 c1(C(C(=O)NCC=C)N(C(CC(=O)OC)C(F)F)C)cc2cccc(Br)c2o1 C1(CNC(=O)C=C2CC2)CCC2CN(C(c3cncc(N4CCCC4)n3)=O)CC12 C1(CNC(c2cnn3c2OCC3)=O)CCCCN(C(=O)Cc2ccsc2)C1 C(CCCOC)(C(=O)N1CCOCC(O)C1)NC(C(F)=CCC)=O C#Cc1cccc(C(N2CCCC(CN(C)Cc3cc(Br)cnc3F)C2)=O)c1.O CC(C)CC(CNC(c1cccnc1C1CC1)=O)NC(C1CC(C)(C)CO1)=O C=C=CCCC(=O)NC1(CNC(=O)C=CC)CCOCC1 c1(C(N2CCN(C)C(CNC(C3CC3F)=O)C2)=O)nnn2c1CSCC2 C1(C(=O)NCC(O)Cn2cccn2)(NC(C=CC(CC)C)=O)CCOCC1 c1(N(C)CC2(C)CC2)nc(NC(=O)OC(C)(C)C)cc(Cl)n1 N1(C(c2ccc(C(N)=O)o2)=O)CCC2CCN(C(C3CC3[N+](=O)[O-])=O)C2C1 c1(C(=O)NC(C(C)C)CCNC(=O)C=CCF)ccc(Cl)c(C#N)n1 C1(C(=O)OC(C2(CN(C)C)CC2)=O)CCC(N(C(=O)CC#N)C)CC1.NC c1(C(C(=O)NCCC2CCCN2C(=O)CCN2CCOCC2)O)ccccc1Cl C1(O)(CNC(C(C2CCC2)OCC)=O)CCN(C(C2CN(C3COC3)C2)=O)CC1 C1(C(=O)NC(C)Cc2cnn(C)c2)(CC)CCCN(C(c2ncccc2C)=O)C1 C12(C(N(CCC)CCNC(=O)C(c3ccccc3Cl)O)=O)CCCC1OCC2 CCCC(CCC)CC(=O)NC1CCC(O)C1.c12ccccc1Cn1cc-2nn1 C(C(CC)CCC1CC1)N(c1nccc(NCC)n1)CC=CC1CC1 c1(C(N(CC(C)CNC(=O)C=Cc2ccncc2)C)=O)ccc(N(C)C)c(F)c1 c1(C(N2CC(NC(=O)CCOC3COC3)C3(C2)CC3)=O)c(Cl)cccc1[N+](=O)[O-] C(=O)(C1=CC2CCC=CCCC12)NCC1N(C(c2cnc(CC)[nH]2)=O)CCCC1 c1(C(C(=O)NCCC(=O)OCC)N(C2CCNC2=O)C)ncc(Cl)cc1F N1(C(c2ccc(NCc3ncn(C)c3)o2)=O)CCCCC1CC(N)=O c1(OC)c(C(=O)NC2CC(O)(CNC(=O)C(O)CN(C)C)C2)c(C)nn1C N1(C(COC(CC)C)=O)CC(C)C(C)(C(=O)N(C)CCF)C1 C1(c2cccc(OC)c2)CN(C(c2ccsc2OC)=O)CCN1C(=O)C(N)=O N1(CC(=O)NCC2(CNC(c3cc(C(N)=O)oc3)=O)CC2)CCCCCC1 n1(CC)cc(CC(=O)NC2(C(F)F)CC(NC(=O)CC(C)N(C)C)C2)nn1 C1(NC(C(CC)n2cncn2)=O)CC(C)CN(C(=O)CNC(c2ccoc2C)=O)C1 c1(CCC(N2CC(N(C)C(c3csnc3Cl)=O)C2)=O)nnc(S)nc1O c1(C(N2CC(C(C)NC(C3(O)CCCCC3)=O)OCC2)=O)ccnc2[nH]ncc12 c1(OC)ccc(N2CC(C(=O)NCC(F)C(C)(C)O)CC2=O)cc1 c1(CCC(=O)NC2(COC)CN(C(C3(O)CCOC3)=O)C2)c(Cl)cccc1Cl c1(C(=O)NCCN(CCC)C(C2CCN(C)C2)=O)cc(Cl)ccc1OC(F)F Cc1cncc(CCC(=O)NC(CNC(=O)CSCC(N)=O)C2CCC2)c1 C1(CC)CN(C(C2(CCF)CCOCC2)=O)CCN1C(=O)CC(C)c1ccco1 C1(CC(N2C3CN(C(C4C(COC)C4)=O)C(C3)C2)=O)CCC2(CCC2)CO1 C(CO)(CN=c1ccc(S(=O)(=O)N(C)Cc2csc(Br)c2)c[nH]1)OC S(=O)(=O)(c1c[nH]c(C(=O)NC)c1)N(CCNC(C1COC(C)(C)O1)=O)CC c1(C(N(C)CC2CCN(C(C3CC3Br)=O)CC2)=O)cc2ccncc2[nH]1 CC1CN(Cc2cnn(C)c2-c2ccc(F)cc2F)CC(C)C1(F)F Cn1cc(Cl)c(CC(=O)N(CC(F)F)CCC2CC2)n1 N1(c2ncc(C)cn2)CC2COCC2(C(=O)Nc2cc(OC(F)F)n[nH]2)C1 Cc1cscc1CNC(=O)CCC1(C)CN(C(C2CCCN2C(N)=O)=O)C1 N1(C(C=C(CCC)C)=O)CCN(C(=O)CC(C)C(F)F)C(c2ccnn2C)C1 Cc1nn(C)c(Cl)c1C(=O)N(C)CCN(C)C(C1CSCN1C)=O C1(NC(c2ccon2)=O)CN(C(C2CCCNS2(=O)=O)=O)C2(CCOCC2)C1 CC1CC(NC(C2CC3(CCC3)C2)=O)CN(C(c2ncoc2Br)=O)C1 N1(C(C2CCN(CC)C2)=O)CCC(C(=O)NCC2CC3CCCC3C2)=C(F)C1 N1(C(C(CCC)C(C)C)=O)CCC2(C1)CN(C(=O)CCNC(N)=O)CCO2 CCC(CC(=O)N1CCN(C(c2cnc(O)c(Cl)c2)=O)CC1CO)CC(F)(F)F C1(NC(CC2N(CC)C(=O)CC2)=O)CCCN(C(=O)CSc2ccccn2)CC1 CC(C)(C)CC(O)CC(=O)NCCCCC(=O)N1CCC(N2CCCC2)C1 c1(C(CNc2c(N(C)C)cccn2)=O)ccc(O)cc1C N1(C(C2CCC(NC(C3CC(SC)C3)=O)CC2)=O)CCC(O)C(C)(C)C1 N1(CC2(C)CNC(=O)C2)CCOCC(C(=O)O)C1 C1(C(N2CC(CNC(c3c(C)n[nH]c3C)=O)C(C(N)=O)C2)=O)OCCCC1(C)C CC1Cc2cc(C(N3CCNCC(O)C3)=O)ccc2N1 Cc1nn(C)c2c(NCCC(=O)N(C)C)nc(=NCC(C)c3ncc[nH]3)[nH]c12 Cc1nccc(C(=O)NCCCCC(C)NC(C2C3CCCOC23)=O)n1 c1(C(=O)NCCC2CCCCN2c2cc(C(F)F)ncn2)ccnc2[nH]cnc12 N1(C(CCc2ncc(C)[nH]2)=O)CC2CC(C1)N(C(C13CCN(CC1)C3)=O)C2 c1(OCCCC)ccc(C(=O)NC2CS(=O)(=O)CC2NC(=O)CC(F)F)c(O)c1 C12(NC(c3c(OC)ccnc3)=O)CCN(C(=O)Cn3nc(C)cc3C)CCC1C2 C=C(Cl)CCC(=O)NC(C1(O)CCCCC1)C(=O)NCC1CC1(C)C Cc1nc(-c2cccs2)[nH]c1C.c12ccc(cc1)s2.C12CCCN1C(=O)NC2C C1(C)(C(=O)NCCC(CC)O)CCN(C(C2CC(CC)C2)=O)CC1 CC1C2CCCCC2CN1C(=O)C(CCF)NC(C1CN(C)CCO1)=O N1(CC2C(C(=O)NCC3(n4nccn4)CC3)CN(CCO)C2)CC2(CCOC2=O)C1 c1(N(C(CC)C)CC)ncnc2c1ncn2C(C)Cc1ccco1 c1(OCC(=O)NC2CC(CCNC(=O)C(F)=C3CCCC3)C2)cccc(Cl)c1 C(=O)(C1CCCc2n[nH]cc21)N1CC(CNC(c2c(C)nns2)=O)C(C)CC1 CC(C)(C)C(O)CC(=O)N1CCC(O)(NC(=O)C(C)(O)C(F)(F)F)CC1 CC1NC(=O)C2=C1N(CCCCCCCS(N)(=O)=O)C(=O)NC2c1ccoc1 N1(C(=O)OC(C)(C)C)CC(O)(C(N2CCC2)=O)C1.c1(O)ccccc1 c1(C(=O)NCC2(C(=O)Nc3c(OC)cccn3)CC2)ccc2cccnc2c1 N1(C(C(C)C2CCC2)=O)CCS(=O)(=O)C(CCNC(c2cccc(O)n2)=O)C1 C1(C(N(CCC(=O)NCCc2cc(C)no2)CC)=O)CCCOCC1 N1(C(C(C)O)=O)CC(C)(C)CC1CNC(=O)Cc1csc(Cl)c1 Cc1cncnc1C(N1CC(SCC(=O)NC2CCCC2)C(F)C1)=O c1(C(=O)OCC)cc(C#N)cnc1NC(C1(F)CCNC1)=O c1(C(=O)NC(CN(C(c2ccn(C3CC3)n2)=O)CC)C)cnn2c1OCC(F)C2 C1(C(C(=O)N(C)CC2C3CN(C(c4c(C)scn4)=O)CC32)O)CCS(=O)(=O)CC1 C1(C)(CNC(C2C(C)CCO2)=O)CCC(NC(C2CC(F)(F)C2)=O)CC1 c1(C(=O)NCC2(CNC(C3C(C)(CC)C3)=O)CCCC2)c(Cl)ccc2c[nH]nc12 c1(C(=O)NC2CCC(NC(C3(CCF)CCC3)=O)C2)cc(O)ncc1F CC1CC(=O)NCCN1C(C1CN(C(=O)C(C)C(F)F)CCO1)=O C1(C(N2CCC(n3cc(CNC)nn3)C2)=O)C2CCCCC12.CC(F)(F)C(=O)O Cc1c(C(N2CCC2CO)=O)[nH]c2cc(C(N3CCC(C)C3)=O)ccc12 C12(CC(=O)NCC(C)(C3CC3)OC)CCC1CN(C(C1CCCN1C)=O)C2 O=C(C(C(F)(F)F)C(F)(F)F)NCCn1cc(-c2ccc(Cl)cc2)nn1 N1(C(c2cc(COC)on2)=O)CC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1 C(=O)(CC(C)CC(F)(F)F)N(CCCNC(c1coc(CO)c1)=O)C(C)C C1(C(N(CCNC(=O)C(C2CCCO2)C2CC2)CC)=O)CC2CCC1CC2 N1(CCC)CCCC1C(=O)NCCCC1CCCN1C(=O)CC1CC1 C(C(F)(C(=O)N1CCC(CCCO)CC1)C(C)C)NC(C1C(C(C)C)C1)=O CC1(C)CCCCC1=CC(=O)NC1CCCC1NC(=O)COCP(C)(C)=O C1(C(N(C)Cc2ccc(Br)s2)=O)COCCN1C(c1cccs1)=O C1(NC(C2CC2C(F)(F)F)=O)CN(C(=O)Cc2nccs2)CC2(CCC2)C1 N1(C(CC2(COC)CC2)=O)CCN(C(=O)CC2CCC(C)(C)CO2)CC1C c1(CC(=O)NC2C=CCN(C(C3C(CC)OCC3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 CC(C)C(O)CC(=O)NC1CCCC(NC(c2cccc(=O)n2C)=O)C1 c1(-n2cc(-c3cc(NC(COC(CC)C)=O)ncc3)nn2)ccc(F)c(C)c1 C(CC(C)C)(C(=O)NCCCC1(CNC(c2cnc(S)n2C)=O)CCCC1)OC C(=O)(C1=C(C)CCOC1)N1CCC2(C(OC(c3c(OC)scc3)=O)C2)C1 CC1CC(C(=O)NCC2CCN(C(c3cnc(C(F)(F)F)cn3)=O)C2)CC(=O)N1 c1(C(=O)NC2CC(CNC(C34C(C)(C)OCC3C4)=O)C2)ccnc2ncccc12 c1(CCC)c(C(=O)NC2(C)CN(C(=O)CN3CCC3C)C2)nnn1C C1(C2CC2)(OC)CN(C(=O)CCCCNC(c2coc(C(N)=O)c2)=O)C1 c1(C(N2CCC(CNC(C(C)OCOC)=O)C2)=O)ccc(Cl)nc1OC c1(C(N2CC(C(=O)NCC(CC#C)(C)C)OCC2)=O)cnc(O)c(C)c1 CCC(C)C(C(=O)N1CCOCC1CC(N(C)CP(C)(C)=O)=O)N(C)C N1(C(c2cc(C)nc(O)c2)=O)CCC(NC(C2(F)CCCCCC2)=O)C(C)(C)C1 N1(C(C(C)(CO)CO)=O)CC(NC(c2cccc(C3CC3)c2)=O)CC(F)(F)C1 C1(C(=O)NC2(C(N(CCN(C)C)CCO)=O)CCC2)CCCC(=O)N1 C(=O)(CC(CC)CCCC)N(CCC(=O)N(CC=C)CCO)C1CC1 c1(CC)ncc(C(=O)NCCC(CNC(=O)CC2C(C)C2(F)F)OC)s1 Cc1cc(C(N2CC3CC3(CNC(=O)CC3C=NN(C)C3=O)C2)=O)oc1C1CC1 C1(NC(C2(c3ccccc3)CC(=O)C2)=O)CN(C(c2cnn[nH]2)=O)CCC1CO N1(C(CC2(C)CCCCC2)=O)CCC(NC(=O)COC2CCOCC2)C(CO)C1 c1(C(N(CC(CNC(C(C)OCCCC)=O)C)C)=O)ccnc(F)c1OC c1(OC)ccc(Cl)c(CC(N2CCC(F)C(NC(C3(CO)CCC3)=O)C2)=O)c1 C1(NC(c2nc(C)[nH]n2)=O)CN(C(c2cccc(OC3CCC3)c2)=O)CC1C C1(C2CCN(c3ncc(C)c(OC)n3)C2)(NC(c2nc(CC)oc2)=O)CC1 C1(C#CC(=O)NC2CC(CNC(=O)COCc3nc[nH]n3)C2(C)C)(CC)CC1 CCC(C)(F)C(=O)NC1CCN(C(=O)CCOc2ccc(CO)cc2)C1 N1(C(C(C)OC)=O)CCN(C(c2ccc(Br)nc2N)=O)CC1C(F)F Cc1onc(-c2ccsc2)c1C(=O)NCC1CC(NC(C2CC(F)(CO)C2)=O)C1 N1(c2cncc(C(=O)OCC)n2)CCCC(C)(C(=O)OC)C1 CCC(CC(=O)N1CCN(C)C(C(=O)N(c2cccc(C)c2)CC)C1)C(C)C c1(C(C(=O)NC2CCC2NC(=O)C(O)c2ccsc2)OC)ccc(F)cc1 c1(C(N2C(C)(C(=O)Nc3cc(Br)ncc3F)CC2)=O)cc(F)c(Cl)c(C#N)c1Cl n1(CC)nnc2cc(C(=O)N(CCN(CC(C)O)C(C3CCSC3)=O)C3CC3)ccc12 N1(C(C=CC2(C)COC2)=O)CC2CCCN(C(=O)C(Cl)=CCl)C2C1 C1(CN(C(Cc2ccc(OC)cc2)C)C=O)CCC(=O)N(C)C1 N1(C(c2c(C(C)O)cccc2)=O)CC(NC(c2ccnc(CO)c2)=O)C2(CC2)C1 C#CCC(C)C(=O)NCC1CC(NC(=O)CCCN(C)C(C)=O)C1 C(CCC(=O)NOCC(=O)OC)NC(C1CCC(CC)O1)=O c1(OCc2cccc(OC)c2)cnc(F)cc1NC(=O)C(=O)NC1CC1 C1(CC(=O)NCC(C(CC)C)O)C2CCCC2N1C(C1(C(F)(F)F)CC1)=O c1(OC)ccc(CN(C(=O)C(n2cc(-c3ccccn3)nn2)C)CC(C)C)cc1 CC(c1ccsc1)=CC(=O)NCCNC(=O)Cc1cc(C)on1 C(C1COC(C)(C)O1)=CC(N1CC2C(CNC(C(C)OCC3CC3)=O)C2C1)=O c1(C(N2C(C)CC(NC(C=NOC)=O)C2)=O)cc(O)cc(C)c1 c1(CSCC(=O)NCC(CO)NC(C2CCCO2)=O)ccccn1 Cc1nn(C)c(C)c1CNC(C1CC(C)(NC(=O)CN2CCCCCC2)C1)=O C1(O)(C(=O)NC(C(=O)OC)CO)CCN(C(=O)COC(C)=O)CC1.C(C)(C)O Cc1ccc(NC(N2CCC(C)(c3cccc(Cl)c3)CC2)=O)cc1Cl C1(c2n(CC3(C)CCC3)nc(-c3ccoc3)n2)CCc2nc[nH]c2C1 CC#CCC(CO)NC(=O)CC(O)CNC(=O)CC1(n2cncn2)CC1 CC1(NC(c2n[nH]cc2Cl)=O)CCCCC1C(=O)NCC(O)C(N)=O c1(C(N(C2CCN(C(Cc3n(C)ncc3Cl)=O)C2)CCO)=O)cc(Cl)c(F)cc1N O(NC(=O)CC(CC(C)C)NC(C1(SC)C=CCC1)=O)CCOCC.OC C1(OC)CCCC1C(N1CC(CNC(C2(CC3CC3)CC2)=O)C1)=O c1(C(N(CCC)CCNC(c2nn(C)c(C)c2Cl)=O)=O)c(C)cc(C)cc1C N(C(=NCCSc1ccc(OCC#C)cc1)NCc1ccns1)CC1CCOC1 N(C1CCCc2n[nH]cc21)C(C1C(CC)CCN1C(=O)C=C(C)C(F)F)=O c1(CNC(c2nccc(C(=O)OC)c2)=O)cc(S(=O)(=O)OC)cc(F)c1Cl CCCC(C)C(=O)NCCN1CCCC(C(=O)NC2CC2)C1 C(=O)(C(CNC(=O)CC1CCCC(=O)N1)(CC)CC)N(CC=C)CC Cc1n[nH]c(C)c1CC(=O)NC1(C(=O)NCCC(=O)N(C)C)CC(CO)C1 C1(C(N2CCN(C(c3cc(C)sc3)=O)C(CCO)C2)=O)OC(C)(C)OC1(C)C C=CC1(C(=O)NC2(C(N3CC(N4CC(F)C4)C3)=O)CCCCC2)CCCCC1 N1(C(CN(C(c2cc[nH]c2)=O)CC)=O)CCC12CCCSC2 C1(C(N2CCC(C(C)CO)CC2)=O)CN(C)CCN1C(=O)C(O)C1CCCC1 c1(C(N2C(C)(CNC(C(C(C)C)(C)O)=O)CCC2)=O)ccc2c(c1)N(C)CC2 N12CC(C)CN(C(C)C1)CC2=O.c1(OC)ccccc1Sc1nccnc1C N1(C(C(C2CCOC2)OCC)C(=O)NC2COC2)CCC(F)(COC)CC1 C(=O)(C(C)(C)N(n1cc(CO)nn1)C)NCCC c1(C(N(CCCNC(C2(C)CCCNC2=O)=O)C)=O)cn(CCO)c(=O)nc1O C1(COC)CC(CNC(c2cn(CCCF)nn2)=O)N(C(c2n[nH]c(C)n2)=O)C1 C(=O)(C(C)(C)CCNC(c1ccc(OC)nn1)=O)NC1(C#C)CC1 C1(CCC(N2C(C)CCC2)=O)CCCN(C(c2nnsc2N)=O)C1 N1(C(Cn2c(C)cc(=O)o2)=O)CCC(F)C(NC(=O)CSS(C)(=O)=O)C1 C(N=c1[nH]c2ncc(Br)cc2o1)c1cc(CC)[nH]n1 CC(CNC(=O)Nc1ccc(-c2cc[nH]n2)nc1)(CO)CC(=O)O c1(NC2C(OC)CN(C(=O)CNC(=O)C3CC3)C2)cccc(Cl)c1N n1(CCCC)cc(NC(=O)N(C2(OC)CCOC2)C)c(C(=O)OC)n1 C1(C(=O)NC(CC=C)(C)C)CCCN(C(=O)CC(C)(C)OC)CC1 C(CN=c1[nH]c(=N)[nH]c(=NC2CCCN3CCSCC23)[nH]1)C1(C)CC1 c1(CNC(c2c(F)cccc2I)=O)ccc(Cl)c(Br)c1 CC1(C)CN(C(C2CC23CC(NC(=O)COC2CCCOC2)C3)=O)C12CCC2 c1(OC)ccc(CCC(=O)NC2CCCN(C(=O)C(C)C3CC3)C2C)cc1C CCC(CC(C)C)C(=O)N1CCN(C(c2cc3c([nH]2)CCCC3)=O)CC1 C(C(CCOC)NC(=O)CNC(c1ccc(Cl)s1)=O)NC(CC1(CC)CCC1)=O C(=O)(CCc1ncc[nH]1)NCCN(C(C1CC1(C)C(F)F)=O)CC N1(C(CC(CC)C(C)C)=O)CCC2C(CCCN2C(=O)Cn2cccnc2=O)C1 C1(C(N(CC(O)CO)CC)=O)CCN(C(=O)CC2(COC)CC2)C1 C12(CCN(C(c3cc(C4CC4)ns3)=O)C1)NC(=O)C(=O)NC2.CC(C)(C)C c1(C(=O)OC(C2C3CCN(CC(F)F)CC23)=O)n[nH]c2c1CN(CC)CC2 Cc1cccc(NC(=O)C(=O)NCC(F)CNC(c2cnncc2C)=O)c1 C1(CC)CCN(C(C2CC(C(=O)OC)C(O)C2)=O)CC1.C(=O)(C(CC)N(C)C)N CCCC(C)CC(=O)N1CC(F)CC1C(=O)NCCC1CCCCC1 CC(C(=O)N1CCCC(CCNC(C2CCCN2C(=O)C(F)(F)F)=O)C1)C(C)O C1(C)(C(N(CCOCCN(C(c2c(CC)cco2)=O)C)C)=O)CC2CCC(C1)S2 N1(C(C2(NC(C(C)SC(C)C)=O)CCN(C)C2)=O)CC2CCCC(O)C2C1 c1(C(N2CC(C)C(NCc3cc(Cl)ncc3Cl)C2)=O)ccc(Cl)c(F)c1F C1(NC(c2cccc3cncn23)=O)CCC2(CCCOC2)C1 c1(-c2cc(C)[nH]n2)ccc2c(C(=O)NCc3cc(Cl)ccc3F)c[nH]c2c1 N1(CCN(C2CCCC2F)C(=O)NC(CC)(C2CC2)C2CC2)CCCOCC1 c1(OC)cccnc1C(=O)NCC1(C(C)NC(=O)Cc2cc(C)on2)CC1.C1(C)CC1 c1(C(=O)OC)cccc(CC(=O)NCc2ccccc2CN=[N+]=[N-])c1 C1(C(N(C)CC2(O)CN(C(C(CCSC)OC)=O)C2)=O)CC2(CCC2OC)C1 n1(CC)ccc(C(N2CCCC(Nc3cc(NC)ncn3)C2)=O)cc1=O C1(NC(C(C(C)C)F)=O)CCN(C(c2ccc(O)cc2)=O)CC1CO C=C(C)CCC(=O)N1CCCC(N(C)C(c2csc(-c3ccc(C)o3)n2)=O)C1 c1(C(=O)NCC=CCNC(C2(C)CCCS2(=O)=O)=O)cc2c(s1)CCOC2 CCCCC(C)CC(=O)NC(CNC(c1ccc(OCCOC)cc1)=O)CC CC(c1ccccc1)=CC(=O)N(CCCOCCNC(=O)C1=CCC1)C Cc1nc(C(=O)NCC2COC(CNC(c3cn(C)ccc3=O)=O)C2)cc(O)n1 CC(CCC(=O)N1CC2CC2(NC(=O)C(CCC=O)OC(C)(C)C)C1)N(C)C C1(NC(CCOCCCOC)=O)CCCCN(C(c2n[nH]c(=N)s2)=O)C1 Cc1nccc(C(=O)NC2CN(C(=O)C=Cc3ccc(C)o3)CC2C)n1 N#Cc1cn[nH]c1C(=O)NCCSCc1cn(CC2CCCO2)nn1 Cn1cc(C2=NOC(C(N3CC(NC(C4CSCCS4)=O)C(C)(C)C3)=O)C2)cn1 CC1(C)CC(=O)N(CC(=O)NC2CCC(NC(c3ncccn3)=O)C2)O1 N1(C(C(OC)OC)=O)CC2C(CNC(=O)C(C)CC=Cc3ccccc3)C2C1 c1(C(=O)NC2CC2C(F)F)cnn2c1SCC2.C12CC1CNC2=O C1(F)(CNC(C(C)(F)c2ccccc2)=O)CCN(C(=O)CCc2ccon2)CC1 N1(C(C2OCC(C)C2)=O)CCCC2(CC(NC(=O)CCC3CC(C)(C)CO3)C2)C1 N1(C(CCC#C)=O)CCCCC1CNC(=O)CCCC1CCOCC1 n1(CC)cc(C(=O)NCC(C)CNC(=O)C(C)n2cccc2)c(C)n1 CCC1=C(C(=O)N2CC(C)(C(=O)NCc3c(F)cncc3F)C2)CCCO1 C(=O)(CCCC(=O)NCC1OCCC1C(=O)NC1CCOC1C)OCC CC(O)CC(=O)N(CC(C)NC(C1CN(C(=O)CC(C)NC(N)=O)C1)=O)C C(CCC1CC1)(C(=O)O)N1CCCN(C)C1=O.CC(O)CC(C)(C)C N1(C(C2(CC#C)CCCCC2)=O)C2CCC1C(CNC(C1CC(OCC)C1)=O)C2 c1(OCCC)cc(C)nc(Nc2ccc(-c3n(CCOC)nc(C)c3)cc2C)n1 N1(C(=O)Cc2ccc(O)cc2)CCN(C(c2cscn2)=O)C2CC12 C(CS(=O)(=O)c1ccc(C)cc1)NC(c1ncc(N(C)CC)nc1)=O C(=O)(CC1CCc2ccc(O)cc21)NCC1CCN(C(C(C)=O)=O)C1 C(CC1=CCC2CC1C2(C)C)N1C(CCc2c(C)cccc2)CCC1 C1(CNC(=NCC=C)NCC2CCCO2)Cc2ccccc2O1 N1(C(=O)CCBr)CCOCC2(C1)CN(C(c1cc3ccoc3s1)=O)CCCO2 CC1(C)C(C(=O)NCC23CCC(NC(=O)CNC=O)(CO2)C3)CC1(F)F N1(C(C2CC=CC(OC)C2)=O)CC2(CC2)CC1C(N1CCCC12CC2)=O Cn1ncc(C(=O)NC2CC(NC(=O)CNC(C3CCCC3)=O)C2)c1N c1(C(=O)NCC(C2CC2)NC(C2(N(C)C)CCCC2)=O)cc(C#N)ccc1N C1(NC(C2CCCC(C3CC3)O2)=O)CN(C(C2(C3CC3)CC2)=O)CCC12CCC2 C1(NC(C2C(C)(C)CC2)=O)CN(c2ncc([N+](=O)[O-])cc2F)CCC12CCC2 c1(C(N2CC3CCCC(C2)N3C(C2CC(F)C2)=O)=O)cnc(O)c2ccccc12 CCCC(C(=O)N(C1CC(CCn2cc(-c3nccs3)nn2)C1)CC)S(N)(=O)=O C#CC1CN(C(C2C=CCN2C(C2(C)CCOCC2)=O)=O)CC1OC c1(C(N2C(CC)CN(C(C3(CC4CCC4)CC3)=O)CC2)=O)cc(C)c(Cl)cc1F N1(C(c2csc(C)c2C)=O)CCC(CCNC(c2nocc2Cl)=O)CC1C C1(C(=O)NCc2cc(Br)ncc2Br)CN(C(=O)Cc2ccccc2)CC1(F)F c1(C(=O)NCC2(Nc3sc(C#N)c(Cl)n3)CCC2)cc2c(cn1)CCCC2 CC(C)C(C(=O)NCC1CCCN(C(=O)Cc2ccc(O)cc2)C1)C(C)C Cc1c(C(N2CCCC2CNC(C2(O)CC(C)(C)C2)=O)=O)nn2ccccc12 c1(C(N2CCCCC(SC)C2)C(=O)NCC(F)F)cc2n(n1)CCCO2 c1(C(N2CCC(N(C(C3CC(=O)N(C4CC4)C3)=O)CC)C2)=O)ccnc(Cl)c1Cl C12CCCN(C1)C(=O)c1sccc1C(=O)OCC(=O)N2CC.C=CCCOCC N1(C(c2n(CC)ncc2)=O)CCCC(CCNC(=O)CC(C)(C)O)C1 c1(SC)cnn(C)c1C(=O)NCC(C)NC(=O)C=Cc1cnc[nH]1 c1(CC(=O)NCc2ccc(C(=O)O)o2)csc(=NCc2ccncc2F)[nH]1 C1(N(C(c2c(CC)ncs2)=O)C)CCCC2CN(C(C3CCCOCC3)=O)CC12 c1(C(=O)NC(c2cccc(Cl)n2)CC)cccc(Cc2cccnc2)c1 C1(N(C)C(C2CC2C(F)(F)F)=O)CCN(Cc2cccs2)CC1 C1(C(N2C3C(NC(c4c(C)occ4)=O)CC(C3)C2)=O)CN(S(=O)(=O)N(C)C)C1 N1(C(c2c(C)sc(Cl)n2)=O)CCC(C)N(C(C23CC(C2)C3)=O)CC1 c1(CNC(Cc2c(C)non2)=O)cc(O)nc(CNC(C2C=CC(CO)C2)=O)n1 Cc1ncnc(C)c1C(=O)NC1CN(C(=O)COc2ccc(F)c(Cl)c2)CC1O N1(C(C2CCN(C(C3=C(C)OCC3)=O)C2)=O)CC2(CCCCCO2)C1 Cc1ccncc1CC(=O)N(CCCNC(c1ocnc1C1CC1)=O)CCO N12CCOC(C1)C(=O)Nc1c(c[nH]n1)C2=O.C1(NC2CC2)CN(c2nncs2)C1 C(=O)(C(F)(F)C(C)O)NCC(C)N(C(c1ccn(CC)n1)=O)CC CCCC(CC)C(=O)N1CCN(C(=O)Cc2cccnc2)CC1COC N1(C(C(CN(C)C)NC(=O)Cc2ccon2)=O)CC2CCCCC2C1 c1(CNC(C2(CNC(C)=O)CCCC2)=O)ncc(C)cc1[N+](=O)[O-] Cc1cn2cc(C(=O)NC3COCC3NC(=O)CSc3ccccc3)sc2n1 C1(CC)CCN(C(=O)CC23CCC(CC2)C3)C1C(=O)NCC1CNC(=O)O1 CCCC(CC)C(=O)N1CC(CNC(=O)CSc2nnnn2C2CC2)CCC1C CCCCCCC(CC)C(=O)N1CC2(COC(CNC(=O)CS(=O)CC)C2)C1 C1(C(=O)OCC)CC12CCCN(CCc1cccn1C)C2 CC(CCN=c1nc(-c2ccsc2)cc[nH]1)NC(=O)C(C)n1cccn1 Cc1cc(C(F)(F)F)cc(NNC(=O)c2ccc(C(C)(F)F)cc2)c1 c1(C(N(C2CCN(C(CNC(=O)OCC=C)=O)C2)C2CC2)=O)cccc2ccoc12 C1(C(C)NC(C(c2ccccc2)OC)=O)CCN(C(=O)C=Cc2cc[nH]n2)C1 c1(C(N2CC(CNC(COCC(=O)NC)=O)C2)=O)sc(=N)[nH]c1C(C)(C)C C(CCCN=C(NCCC1(O)CCOC1)NCC(F)F)SC C1(NC(c2cc3cccnc3s2)=O)C2COCC1CN(C(c1coc(O)n1)=O)C2 C1(NC(c2cncc(F)c2)=O)C2CC3C(C2)C13C(=O)NC1CC12CCCCC2 N1(C(=O)NCc2ccn(CC)n2)CCC(CS)CC1.C(=O)(NC)OC c1(OC)ccc2c(c1)CCC(C(=O)NC1CCC(C(=O)Nc3cncnc3)C1)C2 N1(C(CC(CCC)C)=O)CCC2(CCC(NC(=O)CN3C(=O)CCCC3=O)C2)C1 c1(C(C)C)nn(C)cc1C(=O)NCC1CN(C(=O)CC2CC2(Cl)Cl)CC1O Cn1c(C(N2CCC(CNC(c3c(F)cc(N)cc3F)=O)C2)=O)cc2occc12 CCCCCCC(=O)NC1(CCNC(c2ccn(C3CCC3)n2)=O)CC1 C=CCCCCCCCCCNCc1csc(S(N)(=O)=O)c1 C1(CNC(C2(C(=O)NC)CC2)=O)CCCCC1NC(=O)Cc1ccc(Cl)cn1 C1(NC(CC(=C)Br)=O)CN(C(=O)CC2CCN(C)CC2)C2(CCCC2)C1 C(=O)(C#CC1CCOC1)NC(C)(C)CCNC(c1cnc2n1CCS2)=O C(=O)(C(CC(C)C)OCC)N(c1cn(CC=C)nc1)CCCC.c1cncc(Cl)n1 C1(CCNC(=O)C=Cc2cocn2)CCCCN1C(=O)C(=C1CCCCCC1)F C1(CNC(C23OCC(CC)(C2)C3)=O)CCN(C(c2cn(C(C)C)cn2)=O)C1(C)C C1(C(N2C(CCC(=O)N(CCCF)C)CCC2)=O)(CO)CC(C)(C)C1 N1(C(C2OCCN(C(C(CCC(C)C)O)=O)CC2)=O)CC=C(C(C)(C)C)CC1 C#CCCCCC(=O)NCC(C1CC1)NC(=O)CCNC(=O)CC(C)C c1(C(N2CCCC(N(C(=O)C=C(C3CC3)C3CC3)C)C2)=O)ccc2cc[nH]c2n1 C1(N(C)C(c2cc(C3CC3)on2)=O)CCCC(N(C(=O)Cc2ccsc2Cl)C)C1 c1(C(=O)NC2(CNC(C3CC(C(=O)OC)C3)=O)CCC2)ccc(COC)cc1 N#Cc1ncn(CC(=O)N(CCCc2nncs2)Cc2ccccc2)n1 C(=O)(C(C)CC(N)=O)N1CC2C(CNC(C3(CC=C)CC=CC3)=O)(C2)C1 CCCC(C#N)C(=O)N1CC2C(CN(C)C(c3cc(Br)cn3C)=O)C2C1 C1(N(C(C(C)OC)=O)C)CCCC1(C)CNC(=O)CCc1cnc(C2CC2)o1 N1(C(C(CC)n2cccn2)=O)CC2(CCN(C(=O)COC3CC3)C2)C1 C#CC1(O)CC(C(N2C(C(=O)NCC3COCC(C)O3)CC2C)=O)C1 S(=O)(=O)(CC(F)(F)F)NC1CC(CC(=O)Nc2nc(C)c(I)s2)C1 CCC(C)CN=c1[nH]c(N2CCN(S(C)(=O)=O)C(C)C2)nc2cc[nH]c12 N1(C(CC=C)=O)CCCC(C2CCN(C(c3cnc(CC)nc3C)=O)CC2)C1 C1(C(=O)NCC2OCCN(C(c3on(C)c(=O)c3)=O)C2)COc2ccccc2C1 Cc1cc(N2CC(F)CC2CNC(C2(C(C)C)CC2)=O)ncc1C#N C(=O)(CC(F)(F)C(F)(F)F)NC1(CNC(c2c(N)ccc(OC)c2)=O)CC1 C(=O)(C1CCCc2sc(=N)[nH]c21)N1C(CNC(CCSC)=O)C(C)(C)CCC1 C(C)(C(=O)NCCN(C(=O)C(C)NC(=O)Cn1cnnn1)C1CC1)OC c1(C2N(C(C)=O)CCCC2)ccc(NC(C)CNC(=O)OC(C)(C)C)cn1 c1(N(C)C)ccc(CCC(=O)NCC2(C)CCCN2C(=O)CCS(C)=O)cn1 c1(OCCN(CC)CC)cc(C(=O)NCCC(=O)OC)cc(Br)c1 C1(CCNC(COCCC)=O)C(C)CCCN1C(c1cnc(CO)nc1C)=O N1(C(CC(OCC)OCC)=O)CCC(NC(=O)C=CCSC)C(C)C1 c1(CNC(C2C=CCN2C(C2CC2C2CC2)=O)=O)cccc(C(F)(F)F)c1 c1(C(N2CC(CC=C)(C(=O)NCC(C)(CC)CO)C2)=O)cc(C)nc(C)c1 c1(C(=O)NCCCn2cc(CNC(C)=O)nn2)ccc2c(c1)N(C)C(=O)C2 C1(NC(C(C)(C)n2cncn2)=O)CC2CC1CN(C(C1CC1F)=O)C2 Cc1cc(Cl)nc(N)c1C(=O)NCC1CCCC1NC(=O)COC(C)C c1(CCC2CCN(C(C3CC3NCC)=O)CC2)nccc(C#N)c1[N+](=O)[O-] C(=O)(CC(C)C(C)C)N(C1CCN(C(c2cc(Br)cn2C)=O)C1)CC N1(C(CNC(c2c(C)[nH]cc2)=O)=O)CCN(C(C2C(C)C2C)=O)CC1 N1(C(C23COCC2C3)=O)CCCC(F)CC1.c12cnn(c1)CCNC2=O CC1(C)CN(C(=O)C2=NOCC2)CC2(CN(C(C34CC3COC4(C)C)=O)C2)O1 c1(C(N2CCCCC(NC(=O)Cc3ccc(O)nc3)C2)=O)ccc(F)c(Cl)c1F c1(CC)cnc(C#N)c(-c2cnn(CNCc3cccc(CO)c3)c2)c1 N1(C(Cc2c(C(C)C)cccc2)=O)CCC12CN(C(C1C(C)C1C)=O)C2 C(=O)(C1=NOC2(CCC2)C1)NCC(C(=O)NCc1ccc(OC)nc1)CC(C)C CCCC(C(=O)N1CC2CCCN(c3nccc(C(F)(F)F)n3)C2C1)S(N)(=O)=O C(c1ccc(O)c(O)c1)=CC(=O)N(C)CCN(C)C(c1csc(CO)n1)=O c1(C(=O)NCCC2N(C(C(CC)(C)C)=O)CCCC2)cccn(C2CCC2)c1=O C1(CNC(C2(CCC)CCC2)=O)CCCC(CNC(C23CC(F)(C2)C3)=O)C1 C(=O)(CC(C)(O)C1CC1)NC(C)CNC(=O)CCc1ccccn1 C1(C(=O)NCC2CCCN2C(=O)NC(C2C(Cl)(Cl)C23CC3)=O)(CC)CCSCC1 c1(C=O)cc[nH]c2nccc1-2.C1(C(=O)NC)C=CC(NC(c2occc2CO)=O)C1 C1(C2CC2)(C(=O)NC2C(CNC(c3c(C)scc3)=O)CCC2)CC=CC1 c1(CC)cnn2c1CN(C(c1ccc3c(c1)ncn3C)C(=O)NC(C)C)CC2 Cc1nc(C(F)(F)F)ccc1COC(C)(C)C.C1(=O)C(Cc2nonc2C)O1 CCC(C(=O)NC1CC(NC(c2ccc(C#N)cc2C)=O)C1)C(F)(F)F N1(C(c2c(C)n(CC(C)(C)O)nc2)=O)CC(NC(=O)C(F)C(C)C)C(C)(C)C1 Cn1cnc2c(N3CCC(C4CCOC4)CC3)nc(N3CCC(C)(CO)C3)nc12 N1(C(c2c(C)occ2)=O)CC(C(N2CCC(C)C(O)C2)=O)C(F)(F)C1 N1(C(CNC(C2C(C)CC2C)=O)=O)CCN(C(c2ncccc2Cl)=O)CC1 N1(C(c2cn(CC)nc2)=O)CCC(C(=O)NC2CC(N3CCCC3)C2)=C(F)C1 C1(NC(c2n(CC)ncn2)=O)CC2CC1CN(C(=O)CCc1ccccc1F)C2 c1(C(N2C(CNC(=O)Cc3ccno3)COCC2)=O)cncc2nc[nH]c12 c1(CC)c(Cl)c(C(=O)NCCOCCNC(C23C=CC(CC2)C3)=O)nn1C C1(C(=O)NC(CNC(=O)C(c2ccccc2)O)CO)CC2COCC(C1)C2 c1(C(N2CC(C(C)O)(CNC(C3CC(=O)NC3)=O)C2)=O)ccc2sncc2c1 N1(C(C)C)CCN(C(C(=O)NCC2CC2)C2CCC2C(F)(F)F)C(C)C1 c1(C(N2CCC(NC(c3cnc(C)o3)=O)C(F)C2)=O)cncc2ccc(F)cc12 C1(C(=O)OC)CCC(C)(C)CN1C(C1CCN1C(C)(C)C)=O Cc1cnc(C(N2CCC(C(N3CC(CO)C3)=O)C2C)=O)cn1 c1(C(=O)NC2CN(C(c3[nH]cc(C)c3)=O)C2)cnn(CC(C)C)c1C C12(C(N3CCC(CCC)C3)=O)CCCC1CCN2C(c1cc(C)c[nH]1)=O C1(CC=C)(NC(=O)C(O)C=C)CCCN(C(=O)CCc2cncs2)C1 C(=O)(C(C)CCCOC)NCC(CC)(C)CNC(=O)COC c1(C(N2CCOC(CC)C2)C(=O)NCCCC)snc(OC(F)F)c1Cl c1(C(N(CC(O)CNC(C2(C)CCCS2(=O)=O)=O)C)=O)c(F)ccc2[nH]ccc12 c1(C(=O)NCC2C(NC(CC(C)F)=O)CCC2)ccccc1C#N c1(C(C)(C)OC)nc(=NCCCC(C)NC(C2CCCCC2)=O)s[nH]1 c1(SC)ccccc1CC(N1CCC1CNC(=O)CC1(C)CCN(C)C1)=O CC1CCN(C(=O)CN2CCC2)CCN1C(C1CC1c1cccs1)=O C(CCCCC(=O)NCC1COC(CNC(c2cn(C)cn2)=O)C1)OC C(CC(C(=O)N(C)CC1CN(C(c2cc(C)[nH]n2)=O)C1)OC)OC C1(OC)CCCN(c2cc(NC(C)C3CC3)nc(C(F)(F)F)n2)CC1 CC(C)C(C)C(C)CC(=O)N(CCCN(C(=O)C=Cc1ccc(F)cc1Cl)C)C c1(CC(=O)Oc2cccc(Cl)n2)ccc(-c2ccc(OC(F)F)cc2)c(F)c1 N1(C(c2ccnn(C)c2=O)=O)C2CCCC1CN(C(c1c(Cl)cnn1C)=O)C2 C(=O)(CS(=O)(=O)CC(C)C)N(CCCNC(c1c(C)ccc(F)c1)=O)CCO c1(NC)ccccc1C(N1C(C(N2CCCCC2C(C)C)=O)CC1C)=O c1(C(N2CC(NC(C(COC)C)=O)C(O)C2)=O)ccc2nc[nH]c2c1 C(=O)(C1=CN=C2N=CNN2C1)N1CCOCC(NC(c2coc(C(F)F)c2)=O)C1 C1(CNC(CC(CC)(F)F)=O)CC2CCC(C1)N2C(C1COC(C)(C)C1)=O c12ccc(s1)C(=O)C(=O)NC(C1CCC1)CNC2=O.C1(C(F)F)(CC)CC1 C(CC(F)(F)C(C)C)NC(C1CCCCC1OC)(c1n(CCCOC)nnn1)C C(C(CCO)N=c1cc(NCc2nc(C3CC3)cs2)nc(C(C)C)[nH]1)OC CC1CC(NC(N2CCN(c3ncccc3C(=O)C(F)F)CC2C)=O)CC(C)C1 c1(C(=O)NCCC(=C)CNC(=O)C(C)n2ccnc2)cnn(C)c1C C(=O)(C1CCCc2ccccc21)N1CCC(NC(=O)CN2CCS(=O)(=O)CC2)C1 N1(S(CCC)(=O)=O)CCC(C(=O)N(C(C)CNC(C2(O)CCCCC2)=O)C)CC1 N1(C(C2=CC(C)(C)C2)=O)CC2CCN(C(=O)CNS(C)(=O)=O)CC(C2)C1 CCC(CC(=O)N1CC2CC2(CO)C1)N(C)C(c1cnnc(O)c1)=O C1(C(C)NC(C2CC2F)=O)(NCCCNC(COC)=O)CCC1 C1(N(C(=O)C(F)=CCCF)C)CCN(C(c2cn(C(C)(C)C)nn2)=O)C1 C1(NC(CCC#C)=O)CN(C(=O)Cc2cncc(Br)c2)CCC12CCC2 c1(OC(C)C)ccc(C(N2CCC(NC(c3cc[nH]c3C3CC3)=O)C2)=O)cc1 C1(NC(COC(C)=O)=O)CCC2(CC1)CCN(C(c1ccc(Cl)c3cc[nH]c13)=O)C2 Cc1ccnc2sc(C(=O)NC3CN(C(c4ccncn4)=O)CC3(C)C)c(C)c12 C1(C2(O)CCOCC2)(CNC(N2CC3(C2)OCC2CC32)=O)CCC1 c1(C(N(CC(CNC(c2ccc(C=C)cc2)=O)O)C)=O)cc(F)cc2ccoc12 N1(C(c2cc(CC)c(F)cc2)=O)CC2CC(NC(c3cccn3CC)=O)C(C2)C1 C(C(C(F)(F)F)NC(c1nc(-c2cccc(C(F)(F)C(F)F)c2)cs1)=O)N(C)C C1(C(N2CC(NC(C=CC)=O)C(C)CC2)=O)Cc2ccc(OC)nc2N1 c1(C(=O)O)cc(=NCCCCNC(c2cnc3nccn3c2)=O)[nH]cn1 C1(Cl)(C(N2CC(C(N3CCC(OCC4C=CCC4)CC3)=O)C2)=O)CC2CCC1O2 N1(C(CC(CC)C2CC2)=O)CC2(C1)CN(c1nc(CC)nc(C)c1F)C2 Cc1cccc(C(=O)NC2CCCN(C(c3ncccn3)=O)C2)c1Br C1(CC(=O)NC2(CCNC(C(CSC)O)=O)CCC2)OCCC1(C)C C1(NC(C2C(C=C)CC2)=O)CC(CNC(=O)C(CO)N(C)C)CC1O c1(C(=O)NC(CCNC(C=Cc2scc(C)n2)=O)C)ccc(F)c2ccncc12 Cc1ccccc1SCC(=O)NC1CC(COCCO)N(C(=O)CCCC2CCC2)C1 C1(CC(=O)NCc2cccc(NC(COC(CC)C)=O)c2)CCCC2(CCC2)O1 C(=O)(CCC(=O)N(C(C)C(N1CCC(CCO)C1)=O)C1CC1)N(CC)CC N1(CC(C)O)CCCC1CCN(C(=O)C(F)=C1CCC1)C.C(C(N)=O)OCC C1(c2nnnn2C(C)C)(NCc2c(CC)ocn2)CC(C)N(C)C1 c1(OC)c(C)cnc(CC(N2CC(CCn3cc(C4(O)CCC4)nn3)C2)=O)c1C C(CC(C(=O)NC(CC1CC1)C(=O)OCC)NC(c1nonc1C)=O)CC CCC(C)CC(C(=O)NCCn1cnc(C)c1C)NC(c1cccn(C)c1=O)=O N1(C(c2c(C)occ2)=O)CC2CCCN(C(c3cc(CO)c(C)o3)=O)C2C1 c1(C(=O)NCCCNC(CCCCN(C(C)=O)C)=O)nc(C)c(N)cc1C CC1(C)CC(NC(c2cscn2)=O)CN(C(C2COC3(CO)CC2C3)=O)C1 N1(C(C2(C)CCN(C(C3CC(=C)C3)=O)C2)=O)CCC2(C=CCO2)C1 C(CCC(O)C(=O)Nc1cnn(CC(N)=O)c1)NC(CCC=C)=O c1(NC(C(CC#C)NC(c2ccc(C)o2)=O)=O)c(C)ncnc1C NC(=O)CCC(C(=O)N1CCN(CC2CC2)CC1)n1cc(CC2OCCO2)nn1 c1(CC)cncc(C(=O)N(C)CC2COCCN2C(=O)CC2(C)CC2)c1 c1(C(N2CCN(C(Cc3c(C)cco3)=O)C(C)C2C)=O)oc2ccccc2c1C N1(C(C(C)OC)=O)CC2CCC2(CNC(c2sc(Cl)c(Cl)c2C)=O)C1 c1(C(CO)NC(CCc2cc(C)on2)=O)c(Cl)cccc1Cl N1(CC)CCCCC1C(N1CCSC(C(N2CCC(C)(OC(C)C)C2)=O)C1)=O C1(C(N2CCCC(C(N)=O)C2)=O)(CC)CCN(C(C2CCSCC2)=O)C1 O=C1NCCC2CCN(C(C3CN(C(C4CCCS4)=O)CC34CC4)=O)C12 c1(CC2C(C(=O)NCC(C3CCCC3)NC(=O)CC3(O)CC3)C2)ccc(O)cc1 CCCCC(CC)CC(=O)N1CCN(C(=O)C(C)=C2CCCC2)CC1C1CCC1 c1(C(=O)NCCN(C(C(C)OCC#C)=O)C2CCCC2)cc(F)c(C#N)c(F)c1 C(=O)(C1CCCn2cncc21)N1CCN(C(C(C(C)O)(C)C)=O)CC1CCO C1(CNC(C(C=C)(C)C)=O)COCCN(C(c2csc(C(C)=O)n2)=O)C1 c1(OC)ccncc1-c1cn(CC(=O)NC(CCN2CCCC2)C(N)=O)nn1 C(=O)(CCC(=O)C1CC1)N(CC)CC.C12CCC(C1)NC(=O)c1cscc1OC2 N1(C(c2cnc(CC)[nH]2)=O)CCC2CN(C(=O)CCC3CC(C)(C)CO3)C2C1 CCC(CC)C(=O)NC1CCOC(CNC(=O)CCNC2CCCC2)C1 c1(C(N2CCCC(CC=C)(NC(C3CCC(CC)O3)=O)C2)=O)ccc(N=[N+]=[N-])cc1 Cc1cnn(C(C)C)c1C(=O)NCCC(C)NC(C1CC(F)C(=O)N1)=O C1(C(=O)Nc2ccc(OC)cc2C)CC2(CCN1C(=O)Cn1cnnc1O)CC2 Cc1sc(O)nc1C(=O)NC1CCN(C(C2(n3ccnn3)CC2)=O)CC1 Cc1nc([N+](=O)[O-])cn1CC(N1CC(NC(=O)CCCCCF)CC1C)=O c1(CC(=O)NCCC2(NC(c3ccc(O)nn3)=O)CCC2)ccc(Br)c(F)c1 C1(NC(C(C)(C)OCC)=O)CCOCC1C(=O)NCC(CCC)C1CCC1 c1(C(=O)Nc2scc(CNC(C#CC(OCC)O)=O)n2)cc(F)ccc1F.OC c1(C(=O)NC(c2ccccc2F)CNC(=O)CCC2CC2)c[nH]c2ccccc12 Cc1cc(C)c(C(=O)NC2CC2CNC(c2conc2C(C)(C)C)=O)cc1N C(=O)(C(C)(C)C1CCCC1)NCC(CC)N(C)C(C1CCS1(=O)=O)=O CCC(CC(F)F)C(=O)N1CCN(C(=O)CC2CSC2)CC1C(C)C c1(C(=O)NC(CCC)CNC(c2cc(OC)no2)=O)ccccc1C(F)F N1(C(c2c(SCC)nccn2)=O)CCCN(C(=O)C2=CCCCCC2)CC1CO c1(CN2CCCC(C(=O)Nc3cc(C(F)(F)F)ncc3Br)C2)cccc(F)c1Br c1(NC(C2CC(=C)CN2C(=O)CCc2ccc(C)s2)=O)ncc([N+](=O)[O-])cc1I Cc1cccc(C(=O)NCC2CC(F)CN2c2nc(Cl)ncc2Br)c1C(=O)O c1(C(=O)NCC(CCCC)NC(=O)Cn2cnc(C)cc2=O)ccc(O)nc1Cl Cc1nccnc1C(=O)NCC1C2CC1N(C(=O)CCC(=O)C1CC1)C2 Cc1ccc(C(=O)NC(C)(C)CCNC(C2CCC(C3CC3)C2)=O)nc1O C1(C(N2CCC(C#CC)C2)=O)CC2CCCC2N1C(c1occ2c1CCC2)=O Cc1cc(C(=O)NCC(C2CC2)NC(c2cnc(C3CCCO3)s2)=O)c(C)cn1 N1(C(CCOCC)=O)CCC2CCC(NC(c3nnc(CC)s3)=O)C1C2 c1(OC)ccc(F)cc1CCC(=O)NC(C1(O)CCN(C(C2(O)COC2)=O)C1)C CCCC(CC(=O)N(CC(F)Cl)C)NC(=O)C(C)C(C)OC C1(NC(c2ccc(CSC)cc2)=O)CC2CCC1N2C(c1ccc(F)cc1Cl)=O c1(CC)nc2n(n1)CC(N1CCOCC1)CC2.N1C(=NCCCF)NCC2CC12 N1(c2snc(C)c2C)CC2CC1CC2C(N1CCN(C)CC1C)=O O(NC(=O)C(C)(C)C(C)(C)C)C(C(=O)N(CC=C)CCOC)CC(C)C C#Cc1ccccc1NC(c1ccc(F)nc1)(c1nnnn1CC1CCOC1)C CC(C)C(C(=O)NCC(C)NC(=O)C(C)(C)c1ccncc1)c1ccc(Cl)cc1 c1(C(N2CCc3c(n[nH]c3C)C2)C(=O)NC(CC)C)cccc2cnn(C)c12 CC1(C)COCCC1C(N1CC2CC(NC(C3(O)CCSCC3)=O)C2C1)=O C1(NC(c2cc(Br)no2)=O)CN(C(C2Cc3cscc3C2)=O)CC12CCC2 C1(C(=O)NC(C(C)C)(C)CNC(c2ccc(C#N)s2)=O)CC2(COCCO2)C1 C(C(C(=O)N1CCCC1c1ccc(F)cc1)C(C)(C)C)NC(c1n(CC)nnc1)=O c1(N2CCC(NC(C3(C)C=CCC3)=O)C2)ncc(O)cn1 CCC(C)(CO)C(=O)NCCN(CCOC)C(C12CC(C)(C1)OC2C)=O C1(CC(=O)NCC(C(C)C)O)Cn2nc(-c3ccc(F)cc3F)cc2NC1=O c1(C(=O)NCC(C)(CO)NC(C(C)Cn2ccnc2)=O)nccc2ncccc12 c1(C(N(CC(C)NC(C2(CC(C)C)CCCC2)=O)C)=O)cnc(O)c(Cl)c1 C1(C)(CC=C)CN(C(=O)CC2CC(NC(=O)Cc3nocc3C)C2)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(F)(F)CO)[nH]nc2c(=O)n(C)cnc12 C(C)(c1cccc(Cl)c1)=CC(=O)NC1CN(C(c2c(COC)nn[nH]2)=O)CC1C c1(NCC2(O)CN(C(CCc3ccc(C)s3)=O)C2)ncnc2c(Cl)cc(Cl)cc12 C(CCCCC(=O)NC(C1CCN(C(C2(C)CCSCC2)=O)C1)C)OCC CC1(C)CCC(CO)N(C(=O)C(C2(O)CCCCC2)NC(=O)CCC(F)(F)F)C1 Cc1ncccc1C(=O)NCCOC1CN(C(=O)C(n2nccc2C)C)C1 N1(C(c2ccc(SC)o2)=O)CC(NC(=O)C(Cl)=CCl)C(N=[N+]=[N-])C1 C1(C(N(C)CC2CCCCN2C(C2(C#N)CCC2)=O)=O)CC(=O)OC1(C)C c1(C(N(C(c2ccccc2)CNC(C(C)OCC)=O)C)=O)ccc(Cl)cc1NC C#CCCCC(C)C(=O)N1CCC(C(N2CCC23CC(C)(CO)C3)=O)C1CC N1(C(CCc2cccc(C)c2)=O)CCC2(CC1)CC2C(N1CC(F)C1)=O C1(C(=O)NC(c2nccs2)CC)CN(C(c2ccc(N)c(F)c2)=O)C2(CCC2)C1 c1(OC)ccnc(C(=O)NCC2CCN2C(c2nccc(Cl)c2C)=O)c1F c1(C(=O)NC(CNC(CCCC=C)=O)C(C)C(C)C)cc2nc(C)ccc2o1 CC(F)(F)CC(=O)N1CCCCC1c1ccc(CNC(=O)COCCCF)cc1 C12(C(N(C3CC(NC(C4(C5CC5)CCOCC4)=O)C3)C)=O)CCC(=O)N1CCS2 N1(C(COCC)=O)CCCOC(CNC(=O)C(CC(F)F)c2ccc(F)cc2)C1 C1(C(=O)NC(C2(C(=O)NC(C3CCCC3)CCCF)CCC2)=O)CCCSC1 c1(C(N2CC(NC(C(N3CCSCC3)C)=O)C(O)C2)=O)cc([N+](=O)[O-])cnc1O c1(OCCCC)ccc(CNC(=O)NC(C)CC2CC2(Cl)Cl)c(Cl)c1 c1(OC)ccc(C=CC(=O)NCC(C)(C2CC2)NC(=O)COC(C)C)c(C)c1 C(=O)(C(C)(C)CCNC(c1ccnc(CO)c1)=O)NC1(CO)CC(OC)C1 O=C(C1CCCn2cc(CCO)nc21)NCCCNC(C1(CSC2CC2)CC1)=O Cc1nc(C)c(CN2CCC(O)C2)[nH]1.N12CCCC(C1)C(=O)N1CC(C)(C1)C2 C1(C(N2C(C(N)=O)CC2)=O)CC12CCN(C(=O)CCC1CCOC1)CC2 O=C(CC1=CCOCC1)N1CC(C(=O)NCC2CC(O)C(O)C2)(CO)C1 C(=O)(C1=CC2(CCN(C(C3(C)CC=CCC3)=O)C2)C1)NC1(CC(C)(C)C)CC1 Cc1ccc(NC(C2CC(C)(C)C2)c2nnnn2CCCF)cc1Cl c1(C(=O)NCC(CNC(C2(COC)CC2(F)F)=O)C)cn(C)nc1C N1(CCNC(C(C)N(C(C2C(CC)C2)=O)C)=O)CCCCC1 C#CC1(C(=O)NC2CCCCCC2CO)CCN(C(C2CC=C(C)CC2)=O)C1 C12(C(=O)NCCN(CC(F)(F)F)C)CC(C1)C2 N1(C(c2c(CC)cco2)=O)CCC2(CCN(C(C3CCCC(O)C3)=O)CC2)C1 c1(C(CC)N(C(=O)C(N2CCC(n3cc(C(C)O)nn3)C2)=O)C)ccccc1Cl c1(C(C)OC)nc(C(=O)NCC(O)CNC(C2(F)CCCC2)=O)cs1 c1(NC(CN2C(CC)COCC2)=O)cc(N)c(C)cc1C N1(C(c2cncc(OC)c2C)C(=O)NC2CCOC2)CCOCC(C)(C)C1 C(=O)(C(C)(C)C(C)NC(c1cnc[nH]c1=N)=O)NC(C=C)COC N1(C(C(CC)CO)=O)CCC2(CCCN2C(c2cn(C3CC3)cn2)=O)C1 c1(C(=O)NC2C(C)CN(C(C3CCCC(=O)CC3)=O)C2)noc2ccc(F)cc12 c1(C(N2CC3CCN(C(C(CCC)O)=O)CC32)=O)cnc2ccccc2n1 N1(C(=O)Cn2nccn2)CC2CCN(Cc3ccc4cc[nH]c4c3)C2C1 c1(NC(c2ccc(F)c(-c3c[nH]c4cccnc34)n2)=O)cc(Br)cc2cn[nH]c12 CCC(C(=O)N1CC(O)(CNC(c2ccn(C)c2C2CCC2)=O)C1)C(C)C N1(C(c2n(CCOC)ncc2)=O)CC(NC(=O)CC2CC(C(=O)OC)C2)C(F)C1 C1(NC(c2cnc(C(C)(C)C)nc2)=O)COc2ccc([N+](=O)[O-])cc2C1 c1(NC(C2N(Cc3cnc(SC)nc3Cl)CC2)=O)cc(Br)cc([N+](=O)[O-])c1C N1(C(C=CC=CCC)=O)CC2(COC(CNC(=O)C(CC)OC)C2)C1 C(=O)(C1CSc2ccccc21)N(CCNC(C1CCCC12CC2)=O)CC Cc1cc(C(=O)N(C(C)CN(C(=O)CCc2c(C)noc2Cl)C)C)cc(F)c1C C(=O)(C1Cc2ccccc21)N1C(CNC(=O)CC2CCC3CC3C2)CCC1 c1(C(N(C(CNC(C2(CC#C)CCCO2)=O)C)C)=O)ccc(C2(C)CC2)cc1 c1(C(CC=C)NC(=O)CCC2(C)N=N2)ccccc1 C1(C)(CC)CCN1C(=O)C(C)NC(C1CS(=O)(=O)C1)=O CC(CN(C(=O)CN1CCSCC1)C)C(=O)NCC1CC1Cl C1(CCOC)(NC(=O)C(O)C2CCC2)CCN(C(c2sc(C)cc2Cl)=O)C1 C(=O)(CC(C)(C)C)NCCOC1CCN(C(C(C)=CC)=O)C1 C(C1CN(C(C2CC3CSCC(C2)C3)=O)Cc2ccccc21)NC(C(CC)F)=O N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(=O)CSc3ccccc3Cl)CC2C1 c1(C(N2C(C)(CNC(C(C)SCCCC)=O)CCC2)=O)cc2scnc2[nH]1 Cc1c(NC(c2ccco2)C)ncnc1N(C)CCF c1(CNC(C(C2CC(NC(=O)C=Cc3cc[nH]n3)C2)F)=O)ncccc1Cl c1(CNC2CCC(C#C)CC2)cc(C)nc2ncnn12 C1(NC(COCP(C)(C)=O)=O)CCCC(NC(=O)CCc2ccc(N)cn2)C1 CC1COC2(C1)CN(C(c1cnn(-c3ccccc3)c1Cl)=O)C2 Cc1ncc(C(N2CC(n3cc(C4(O)CCCC4)nn3)C2)=O)n1C c1(C(C)NC(=O)OC(C)(C)C)[nH]ccc1NC(N1CCC(O)C1)=O Cn1ncc(C(=O)NCC2CCn3nnnc3C2)c1S(N)(=O)=O C1(N(CCOC)C(c2ccsc2)=O)CCN(C(=O)C(c2c(C)noc2C)C)CC1 c1(C(C)NC(c2cnoc2)=O)ccc(CNC(=O)COc2cccnc2Cl)cc1 O=C(CCCCO)NCC1(F)CC(CNC(=O)CCc2ccc(Cl)nc2)C1 c1(C(N(C(CC)CNC(=O)CCN2CCC(F)C2)C)=O)cncnc1C C1(NC(c2cc(C)on2)=O)CN(C(=O)CN2CCC(C)(C)C2)CCC1CO C1(NC(c2cnc(O)c(F)c2)=O)CC2CC1CC2C(N1CCOC(CCO)C1)=O c1(CNC(COCC)C)ccc(C(F)(F)Cl)cc1 c1(C(C)NC(C2(NC(c3cnc(C)n3C)=O)CC2)=O)cccc(C#N)c1 CCCCC1CC(=O)N(C)CC(C)N1.C1(C(=O)N(C)C)(C(C)(C)NC(C)=O)CC1 c1(C(N2CCC(C(N3CC(C)(C)SCC3)=O)O2)=O)cccc2[nH]ncc12 c1(C(=O)NC2(CCOC)CCN(C(C3C(=C)C3)=O)C2)cnn2c(O)cc(C)nc12 C1(CC=C)(NC(=O)C(=C2CCCCC2)F)CCCN1C(=O)COCCF c1(OC(C(=O)NC(c2ccc(C)cc2)CF)C)cccc(Cl)c1Cl N1(CC)CCCSCC1CNC(c1nc(=O)n(C)[nH]1)=O CCC(CCC(=O)N1CC(NC(c2c(Cl)cnn2C)=O)C(O)C1)OC C1(CNC(c2cn(CCC)nc2)=O)(OC)CCN(C(c2snnc2C(C)C)=O)C1 C(CC(C(=O)N1CCC(C(F)F)C1)OC)NC(C(C)OCC=C)=O Cc1ccc(C(=O)NCC2(NC(c3nccnc3C)=O)CCC2)cc1 CC1(C)COCC1C(=O)NCC1CCN1C(c1cnc(C(F)(F)F)nc1)=O C#Cc1cnn(CC(=O)NCCCC(C)NC(=O)C(CC)SCC)c1 C(=O)(CS(N)(=O)=O)N1CC(O)(C(C)NC(C2CC(C)(C)C2)=O)C1 Nc1nc(C(=O)NC2CC(NC(=O)CC3(CO)CC3)C23CCC3)ccc1[N+](=O)[O-] c1(Cn2ccc(C(N3C(c4ccn(C)n4)CCC3)=O)n2)ccc2c(c1)OCCN2 c1(C(=O)NC(CC=C)CNC(c2csnc2OC)=O)cc(Br)ccc1F N1(C(COCCN(C(=O)C(C)(C)n2cnnn2)C)=O)CCCC1c1cc[nH]n1 C#CCC(CC(=O)N1CCN(CC(C)O)CC1)NC(=O)COCCC(C)C c1(SCCC#N)cccc(OC(F)(F)F)c1.C1(O)(CC=O)CCOC1 C1(F)(CNC(C(C)(C)C2CCOC2)=O)CCCN(C(=O)CCC2CCOC2)C1 Cc1ccc(C(N2CCS(=O)C(C)C2)C(=O)NC(C)C)c(F)c1 c1(OC)cc(C(=O)NCC2CCC(NC(=O)C=C3CC3)C2)cc([N+](=O)[O-])c1O Cc1[nH]nc(CO)c1C(=O)NC1CC2(C1)CC2C(N1CC(N2CCC2)C1)=O C(=O)(C1=C2CCCN=C2NN1)NCC1N(C(c2cccc(C)n2)=O)CC1 C1(C(N(CCN(C(=O)Cc2ccsc2Cl)CC)CC)=O)CCc2cncn2C1 Cc1nn(CC(=O)NC2CC2NC(=O)CC=CC(C)(C)C)c(C)c1Br C1(CNC(C=Cc2n(C)ncc2)=O)CC(NC(=O)CCCC2CCC2)C12CCC2 CC1(C)CN(C(C2CCCC2)=O)CC1NC(=O)Cn1nncc1Br c1(NC(=O)C=Cc2ccc(Cl)nc2)cnc2c(F)c(F)ccc2c1 c1(C(=O)NC2(CCC)CCCN(C(c3nccn3C)=O)C2)ccc2[nH]ccc2c1 c1(NC(C=NCCOC)=O)ccc(CCC(N)=O)cc1.C(C=O)=CCOCC#C C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC1CC(NC(c2c(C)ncnc2C)=O)C1 N1(C(c2n(CC)ncc2)=O)CCC(C)(C)C1CNC(C1(Cl)CC1(F)F)=O c1(C(N2C(C)CCC(NC(C3(CC(C)C)CC3)=O)C2)=O)cccc2cnsc12 N1(CC(=O)NC2COCCN(C(c3c(C)n(C)cn3)=O)C2)C(=O)C(C)C(C)C1=O C1(C(N2CC3C(NC(CC(C)n4cccn4)=O)C(C3)C2)=O)CCN2CCCC2C1 C1(NC(C(C)NC(C)=O)=O)CN(C(c2cc3ncccc3s2)=O)CC(F)(F)C1 N1(C(c2nc(COC)sc2)=O)CCN(C(c2ccc(SC)cc2Cl)=O)C2COCC12 C(=O)(C(C(C)NC(c1cc(COC)[nH]n1)=O)C(C)C)NCCC(CC)(O)CC N1(C(c2cc(C)n(CC(F)(F)F)n2)=O)CCN(C(=O)Cc2ccsc2)CC1CF c1(C(C)C)ccnc(N2CC3CC3(CNC(=O)Cc3ccc(CO)cc3)C2)n1 c1(OC)cnc(Br)cc1C(=O)NCC(C)NC(=O)Cn1ccnc1C C(C)(CNC(C1(c2ccno2)CC1)=O)(C(C)C)NC(C(CC)c1ccccc1)=O C(=O)(C(F)C(F)(F)F)NCC=CCNC(CC1(CC)CCCCO1)=O CC1CNc2c(C(=O)NC(C)(C)CCCNC(C3CCCC3)=O)cccc2C1 c1(C(=O)NCC2CCN(C(c3n(C)ncc3)=O)C2)cc(F)c(C(F)(F)F)c(F)c1 Cc1cc(Br)cc2c1C(NC(=O)C(=O)NC1CC3CCCC3C1)CC2 CCCCC(O)C(C)C(=O)NC(CCCC)CC(=O)N1CCC(C#N)C1 Cc1cn2ccc(C(N3CCCN(C(C4C(C)C4(F)F)=O)C(C)C3)=O)cc2n1 c1(C(=O)NCC2(C)CCCN(C(CC(=O)OC)=O)C2)cc(Cl)c([N+](=O)[O-])[nH]1 N1(C(c2c(CNC(=O)C=CC3CCOCC3)noc2)=O)CC2CC=CC1C2 CCC(O)C(=O)N1CCC(C(C)NC(=O)C(C)(C)N(C)C)C1 C1(NC(=O)CCc2ccoc2)(CO)CCN(C(C23CCC(C2)C3)=O)C1 N1(C(c2n(CC#N)ncc2)=O)CCCCC(NC(c2coc(Br)n2)=O)C1 C1(C(=O)OCC)OCCNCC1N1CCN(c2cccc(C)n2)CC1 C(=O)(CCC(CC)OC)NC1CCC(NC(Cc2c(COC)cccc2)=O)CC1 C(=O)(C1CCCc2c1ncn2C)NCC(CC)NC(c1ccc(C2CC2)nc1)=O Cc1ccc(C(=O)NC2CC(NC(C3(C4CC4)CC3)=O)C2)c(F)c1 C(=O)(C1=CC2CCCC12)NCC12CC(CNC(CC(CC)(F)F)=O)(OC1)C2 C=C1CCC(C(N2CCC2CNC(=O)CSCCC)=O)CC1 c1(C(=O)NCC(CC)NC(c2ccc(F)c(Cl)c2F)=O)cccc2cc[nH]c12 c1(CC(=O)NC(C)C(N)=O)ccc(O)c(CNC(C23C(CN(C(C)=O)C2)C3)=O)c1 C(C(C)(C)C(=O)NCC1CCC(C)N1C)N(C(c1cc(OC)ns1)=O)C N1(C(c2ccc(C(C)C)nc2)=O)CCCC2(C1)CN(C(=O)C(C)(C)C(C)(F)F)C2 C1(C)(CC)CC(NC(c2cncc(F)c2)=O)CN1C(c1sccc1C#N)=O c1(N2C(C)C(NC(c3nccn3C)=O)CCC2)ncnc2c(Br)cccc12 N1(C(C=CC(=O)OCC)=O)CC2CC(NC(=O)Cc3c(OC)noc3CC)C1C2 C1(COC)CN(C(c2cc(Cl)ncc2C)=O)CCN1C(c1ccnc(Cl)c1Cl)=O N1(C(CCCOC)=O)CCN(C)C(C(=O)NC2(C)CCC2)C1 C1(NC(C=CSC)=O)CC2CCC1(NC(=O)C(C)Cc1ccccc1)C2 Cc1cc(=NCCc2nnc(C)s2)[nH]c(=NCC2CCN(S(C)(=O)=O)C2)[nH]1 c1(C(=O)NCC2C(CNC(c3ccc(CC)nc3)=O)C2)cc(F)cc2cc[nH]c12 c1(OCC(=O)N(C2CCC(CNC(C3CC4CC4C3)=O)CC2)C)cccc(C#N)c1 N1(C(C(C)Oc2ccc(SC)cc2)=O)CCC(NC(C2CCC2)=O)CC(C)(C)C1 C1(NC(CSc2cc(C)ncc2)=O)CCC2(C1)CN(C(=O)Cn1ncnn1)C2 C1(C(N2CCCC(C)C2CNC(C2CCC(=O)N2)=O)=O)CC2(CCOCC2)CO1 c1(C(N(C2CCN(C(c3cc(C(F)F)no3)=O)C2)CC)=O)ccccn1 c1(C(=O)NC2CCCN(C(C(c3cccc(O)c3)C)=O)C2)cc(F)ccc1F c1(C(N2C3CCC2C(NC(C2(O)CCCCC2)=O)C3)=O)ccc(Cl)cc1Cl C#Cc1ccc(CNC(=O)N(C2(c3ccccc3)CCC2)C(C)C(C)C)cc1 O=C1CCC(CNC(=O)CCC2CCC(NC(=O)Cn3cnnc3)C2)O1 c1(C(=O)NCC(C(C)(C)C)NC(C2C(=C)C2)=O)ccc(C(=O)NC)c(F)c1 C1(C(=O)NCCOC2CCN(C(Cc3n(C)ccc3)=O)CC2)CCC2(CCC2)C1 c1(OC(c2c(N(C(c3ccc(CC)[nH]3)=O)CCO)c[nH]n2)=O)ccc(Cl)cc1 c1(C(=O)OC)ncoc1C1CCN1C(=O)NCC1(CCC(F)(F)F)CC1 CC(CCCN=c1cc(C2CC2)nc[nH]1)NC(=O)C(C)(C)C1CC1 Cc1cc2nc(C(=O)NCC(C)(C)NC(c3ncc(Cl)cc3F)=O)cn2cc1C c1(C(=O)NCC23C(CN(C(CC4CC(OC)C4)=O)C2)C3)cc(C)ccc1F N1(C(C2(CC=C)CCCC2)=O)C2CCC(C(N3CC(C(N)=O)C3)=O)C1CC2 Cc1nc(C2CC2)n[nH]1.C(=O)(C(C)(c1ccccc1)N)NC1(CNC(CS)=O)CC1 C(C(C)(C)CNC(c1cnn(CC)c1)=O)N(C(c1csnn1)=O)CC c1(C(N2CC3(CC(NC(C4C(CCC)C4)=O)C3)C2)=O)ccnc2c1ccn2C c1(NC2CCCN(C(C=C(C)CCc3ccccc3)=O)C2)cc2nncn2cn1 CCCCC(O)CC(=O)N1CCC(NC(C2(Sc3ccccc3)CC2)=O)C1C c1(OCCCCNC(C2C(C(C)C)OCCC2)=O)cc(Cl)cc(Cl)c1 CCC(CC)CCC(=O)NC(CO)C(C)NC(C1CCC(C(=O)OC)O1)=O N1(C(C=C(C)C(C)(C)C)=O)CC(C)(C)CC1CC(=O)N(CCO)CC1CC1 Cc1c(Cl)ccc(C(N2CCN(C(=O)C(C)C3CCC3)CC(O)C2)=O)c1O C1(C(N(CC(CC)OC)C)=O)CCN(C(=O)Cc2ccc(Cl)c(C)c2)C1(C)C c1(C(=O)NCC2(COC)CN(C(C3(C)CC3F)=O)C2)oc(Br)cc1C C1(NC(C2C(CC)CCC2)=O)CCN(c2ncnc3[nH]ccc23)C12CCCC2 c1(CNC(CCOCC)=O)cnn2c1CN(C(=O)C(C1CCOC1)CC)CC2 C1(NC(=O)NC2(Cl)C(C(C)=O)C2)CCc2nncn2C1 Cc1cccc2[nH]c(C(=O)NCC(F)CNC(c3cn(C)[nH]c3=N)=O)cc12 C1(NC(C2(COC)C=CCN2C(=O)C(O)CN(C)C)=O)CCCN(C)CC1 c1(C(=O)NCC2N(Cc3n(C)ccn3)CCSC2)ccc(F)cc1Br Cc1ccc(C(N2CCC(NC(=O)C(C(C)C)n3cnc(C)c3)C2)=O)c(N)n1 C1(NC(C2N(C(C)C)C(=O)CC2)=O)COC2(CCCN(C(=O)OC(C)(C)C)C2)C1 C(CN=C(NCc1cnc(N(C)C)cn1)NC1CSC1)N1CCCC(OC)C1 N1(C(c2cc(CNC(COCC=C)=O)no2)=O)CC(F)(F)CC1CO C=C(Br)CC(C)(C)C(=O)N1CC(CNC(=O)Cc2ccccc2SCC)C1 Cc1nc(C(=O)N(CCCNC(=O)CN2CCCC2C)CC2CCCC2)co1 c1(OC(C(=O)N(C2(CNC(C(C)OC)=O)CCC2)C2CC2)C)ccc(Cl)c(Cl)c1 Nc1cnc(C(=O)NC2CC23CC(NC(=O)CC2COCCOC2)C3)cn1 C(=O)(C1=CS(=O)CCC1)N1CCC(C)C1CNC(c1cc(F)ccc1Cl)=O c1(N2CC(CNC(COCCOCC)=O)OCC2)ccc(C#N)cc1[N+](=O)[O-] C1(C)(NC(C2C(C)(C)CCC2)=O)CCCN(C(c2cccc(N)c2N)=O)C1 N1(C(C(C)SCc2ccccc2)=O)CC2CC(NC(=O)CC3(CO)CC3)C2C1 CN1N=C(CC(=O)NC23CC2CN(C(c2cc4ccc(Cl)nc4s2)=O)C3)CC1=O c1(C(=O)NCC(CC)NC(C2(CC)CC2(F)F)=O)cc(O)nc(Br)c1 N1(c2cc(NC(CC)CN3CCCC3)ncn2)CCc2cccc(O)c2C1 N1(C(CCc2cnc(C)o2)=O)CCC(C(=O)NCC(C)CCCO)(C(C)C)C1 C1(CNC(C2(CC#C)CCOC2)=O)CC(C)CCN1C(c1ccsc1C#N)=O C(=O)(C1=CS(=O)CCC1)NCC1CC2CN(C(Cn3c(N)ccn3)=O)CC21 Cc1n[nH]c(=NC2CC3CN(C(=O)CCCCC(F)F)CC23)o1 C(=O)(CCCNC(=O)COC1CC1)N(CC(=O)OC(CC)(C)C)C N1(C(C(CC)C)=O)CCC2(CCCC2CNC(C23CC(C2)C3)=O)CC1 C1(CNC(C(C)OCCOC)=O)CCCCN(C(=O)CCCn2cc(C)cn2)C1 CCN=c1cc(-c2nc(C3C(C)(C)C3(F)F)n(-c3ccc(OC)cc3)n2)cc[nH]1 CC1(C)CCN(CCNC2(C)C(=O)C2CC)C1.OC C1(NC(CN(C(CC2CC(=O)NCC2)=O)C2CCC2)=O)CC2(C1)C(F)(F)C21CCC1 C(C(F)(C(=O)NCC12CCC(CC1)O2)C(C)C)NC(c1c(C#C)cnn1C)=O c12cccc(n1)C(C1CC1)c1n(ncc1)CO2.c1(C(=O)OC)ccccc1.C1CC1 c1(CCC(=O)N(CC(CNC(CCSCCC)=O)C)CC)c(F)cccc1F n1(CC)cc(NC(=O)CC2CCCN2C(=O)Cc2ccoc2)c(C(C)(C)OC)n1 c1(SCC)ccc(CC(=O)NC2CCC(C)(CNC(=O)CO)C2)cc1 N1(C(CCC=C)=O)CCC(C)(C)C1CNC(=O)CC(C)SC C(=O)(C(CC(=O)NCC1(NC(C2CCC(C)(C)CC2)=O)CCC1)C(C)=O)OCC C(c1ccccc1Cl)=C(C)C(=O)NC(C1(O)CCN(C(C2CC(=O)C2)=O)C1)C C(=O)(CC(C(=O)NCc1cccc(S(C)=O)c1)C(C)C)OCC C=CC(CCC)CC(=O)N1CCN(CC(C)NC(c2coc(C3CC3)n2)=O)CC1 N1(C(CSCC=C)=O)CCN(C(C2(O)CCOCC2)=O)CC1CO C1(NC(C2(CC#C)CC=CCC2)=O)CN(C(c2n[nH]c(CC)n2)=O)CC1(C)C C1(C(=O)NC(C2(O)CCN(C(=O)CCS(C)=O)C2)C)CC12CCCCCC2 Cc1ccc(CN2CCCC(C(=O)Nc3cccnc3I)CC2)cc1[N+](=O)[O-] C(=O)(CCCC1CC1)NC(C1CN(C(c2cnn(-c3cccs3)n2)=O)C1)C CN1CCCCC1CC(=O)N(C1CCCN(C(c2cnn(C)n2)=O)C1)CC1CC1 C1(C(=O)NCC2(C)CCN(C(=O)CCc3cccnc3F)C2)(OC)CCCOC1 C(C(CC(C)C)C(=O)NC1CCC1C(=O)NC1CC=CC1)OC C1(C(N(C)Cc2c(C)nco2)=O)CN(C(C2(CF)CC2)=O)CC(C)(C)C1 N1(C(COC(C)C)=O)CCC(CNC(c2cccn(C)c2=O)=O)CC1C N1(C(CC(C)c2ccccc2)=O)CC2CC1C2C(N1CC(O)C1)=O CC1(C)CCOC(CNC(C2CC23CCN(C(C2COCOC2)=O)C3)=O)C1 O=S1(=O)c2ccc(c(Br)c2)N1.c1(NCC2CCC2O)cccc(F)c1F C1(C)(C(=O)NCC2(CC)CCCO2)C=CCN1C(c1ccc[n+]([O-])c1)=O C1(C(=O)NC2C(CNC(COC3(C)CCOCC3)=O)C2)CCC2CCCCN12 c1(OC)nc(C)sc1C(=O)NC1(C)CC(NC(c2cccnc2N2CCCC2)=O)C1 c1(OC)ccc(C(=O)NCC2CN(C(=O)C(C)N3CCC3)CCO2)cc1C1CC1 O=C(CC(CC(F)F)C1CCC1)NCC1CCCCN1C(c1occc1F)=O CCCCCC(O)CC(=O)NC(CCCOC)C(=O)NC(C)(C)CCCF C(=O)(C1=NOC(C)(C)C1)NCC1(C(C)(C)C)CCN(C(CSC)=O)C1 C1(S(N)(=O)=O)(C(N(CC(C)NC(c2cccnc2C(F)F)=O)C)=O)CCCC1 c12nccnc1C(=O)N2.N1(C(C2(C)CN(c3nnc(C)o3)C2)=O)C(C)CCC1C C1(C)(C(N2CC(C)(CF)C2)=O)CN(C(C2(O)CCC2)=O)C(C)(C)C1.C1CC1 CCN=c1[nH]c(C)c(C(N2CC(NC(c3c(C)ncnc3C)=O)C(C)C2)=O)s1 C(=O)(C1c2ccccc2C2CC1C2)NCCC(C)NC(=O)CC1CCN(C)C1=O c1(NC(CC)CNC(=O)C(C)(C)CF)cc(C)c([N+](=O)[O-])cc1C#N C(=O)(C1=NN2CCCN=C2N1)NC1CN(C(C(C)N2CCC2)=O)CC(O)C1 C1(C(=O)NCCN(C(=O)CC2(CC)CCC2)CC)Cc2cncn2C(=O)N1 C1(C(=O)NCC)CCCN1C(C1CCC(NC(c2ocnc2C)=O)C1)=O C=CCC(CC=C)C(=O)N(CCC(=O)NCC1(CC)CCOC1)CCO c1(CN2CCC(CC(=O)Nc3cc(Cl)c(F)cc3Br)CC2)ccc(F)c(F)c1Cl c1(CN(CC(C2CCC2)OC)Cc2ccc(I)s2)oc(C(=O)OC)cc1Br c1(C(N2CC(O)(C(=O)NCCN(C3CCCC3)C)C2)=O)cc(C(=O)O)cc(Br)c1 c1(CC(=O)NC2CC3CC(Nc4cncc(Cl)n4)CC3C2)ccc2occc2c1 C(=O)(C1=CS(=O)CCC1)NCC1CC(NC(C(C)OCC(F)(F)F)=O)C1 n1(CC(=O)NCC2CC(NC(C(C)c3ncco3)=O)C2)ccc(=O)n(C)c1=O Cc1ccc(NCc2cnn(CC)c2)c(C)c1 c1(C(N2CC(CNC(=O)CC34CCCC3C4)C(O)C2)=O)cccn2nnnc12 CC(C)CC(C(=O)NCCc1cnn[nH]1)ONC(=O)CCc1nc(O)n[nH]1 c1(C(=O)NCC2N(C(C(CC=C)(C)C)=O)CCC2)c(F)cc([N+](=O)[O-])cc1Br c1(C(N2CCOCC2CNCc2ccc(F)c(O)c2F)=O)ccc(F)c(F)c1F c1(C(N2CC(CCC)N(C(C3CCCS3(=O)=O)=O)CC2)=O)c[nH]c2cccnc12 Cc1nc(N(C2CCN(C(c3cncn3-c3ccccc3)=O)C2)C)cc(C#N)n1 CC1CCN(C(C2(O)CCCCC2)=O)CC1CC(N1CCC2(CSC2)C1)=O Cc1nc(C=CC(=O)N(C)CC2(O)CCN(C(=O)C(O)C(C)(C)C)C2)[nH]c1C C12CC(c3nnnn3C3CC(F)(F)C3)(C1)NCC2.C1(CNS(C)(=O)=O)CCCSC1 c1(-c2ccc(C(=O)OC)nc2)ccc(S(=O)(=O)N2CCCCC2)s1 c1(C(N2CC(C(C(=O)NCCN(CCC)C(C)C)O)C2)=O)ccc(O)cc1 Cc1n[nH]c(C)c1CNC1CCCC1C(=O)NC(C)Cn1cnnc1 c1(C(C(=O)NC(CNC(C2(C(C)C)CCC2)=O)CO)C2CC2)cccc(Cl)c1 CC(CNC(c1cc(C#N)c[nH]1)=O)CC(=O)N1CCN(CC2CC2)CC1 N1(C(C)CC(=O)NCC2CCN(C(C3CC(F)C3)=O)C2)Cc2ccccc2C1=O CC(CCN=c1cc[nH]cc1S(=O)(=O)N1CCCC2(CC1)CC2)N1CCOCC1 c1(OC)c(C(=O)NC(C)Cn2cc(C3CCCN3C)nn2)cccc1F N1(C(CC2CC(C)(C)OC2)=O)CC(CO)C2(C1)CN(C(C1CS(=O)(=O)C1)=O)C2 CC1(C(=O)NC2CCCCC2n2cc(C(=O)NC3CC3)nn2)CCCNC1=O Cc1cccnc1C(F)(F)C(=O)NCC(C)(C)CN(C)C(c1cnc(S)nc1)=O CC1OCCC1(O)NC(=O)NC(=O)OC(C)(C)C.c12cccc(c1)NC(=O)N2.C(C)(C)O C1(NC(CCN(CCCO)C(C)=O)=O)CCC2(CC1)N=N2 c1(C(N2CC(NC(C34CC(C3)C4)=O)CC(F)(F)C2)=O)ccc2ccsc2c1 N1(C(c2c(CC)cco2)=O)CCC2(CC1)CC2C(=O)NC1(CC)CC=CCC1 n1(CCC)nc(C)c(C(=O)NC2CCCCN(C(=O)CC3C=CCCC3)C2)c1C CC(C)C(C)C(=O)N1CC(CNC(C2(C(C)(C)C)CCCC2)=O)(COC)C1 C1(C(=O)NC(Cc2ccc(CNC(C(CC)C#N)=O)cc2)C)CN2CCN1CC2 C1(C(C)NC(c2cnn(C3CCCC3)c2)=O)CN(C(C2CCC2)=O)CCO1 Cc1cccc2c(C(=O)N(CCN(C(=O)C(F)C3CC3)C)C(C)C)nccc12 CCCCC(C(=O)NC12COC(C1)C(NC(C1CC(OC)C1)=O)C2)OC CC(C)CC(CNC(=O)COC1CC=CC1)NC(C1CCCC(C(N)=O)C1)=O c1(C(=O)OCC)cc(CN(C)C(c2cnc[nH]c2=N)=O)nn1C C1(C(N2C3CC(NC(c4c(C)snn4)=O)C(C3)C2)=O)CN2CCN1C(C)C2 CC1=NOC(C(=O)NCC(C)N(C(COCCCC)=O)CC)C1 c1(C(N(CCC(=O)N2CC(C(=O)OC)C2)CC)=O)c[nH]c(=O)cn1 C(=O)(C1=C(Cl)CCC1)NCCCCN(C)C1CC1.C12(OC)CN(C1)C(=O)C2 N1(C(C=CCCC)=O)CC(C)C(C)(CNC(=O)CN2CCC(C)C2)C1 C1(C(=O)NCCN(CCC)C(c2cccc(OC(F)F)n2)=O)CC(=O)N(O)C1 C1(C2CN(C(=O)CC3CCC4CC4C3)C2)(NC(c2ccc(CO)cc2F)=O)CC1 C1(CN(C(=O)CSC(F)F)CC)CCCCN1C(c1cnc(C(C)=O)s1)=O C1(CNC(C2C(CN=[N+]=[N-])C2)=O)CCCCC1CNC(c1sccc1CO)=O C1(O)(CNC(CN(C(CNC(CC)=O)=O)C(C)C)=O)CCC(C)(C)C1 C1(C(=O)NCC2CC(NC(c3c(C)ncnc3O)=O)C2)CC12CCC(C)(C)CC2 c1(C(=O)NC2C(NC(=O)CCSc3cncc(F)c3)CC2)cnc2nccn2c1 N1(C(=O)NC(CC)(CC)CC(F)(F)F)CCC2(CCN(C)C2=O)C1 N1(C(c2[nH]cc(C)c2)=O)CCCN(C(c2ccc(F)cc2C2CC2)=O)CC1C c1(CNCC2CCCCC(NC(=O)OC(C)(C)C)C2)cccc2c1CCOC2 C1(NC(c2c[nH]nc2-c2ccc(Cl)cc2)=O)CN(C(C2(CCF)CC2)=O)CC1F CC1CN(C(=O)Cc2ccsc2)CCN1C(=O)CNC(S(=O)(=O)C1CC1)=O N1(C(Cc2c(C)n[nH]c2C)=O)CC2OCC(NC(=O)C=Cc3ccccc3)C2C1 c1(N2CCC(CC#C)C2)ccc2nnc(Cn3cc(C)cn3)n2n1 Cc1noc(C)c1S(=O)(=O)N1CCc2cc(-c3c(F)ccc4occc34)ccc21 C1(c2n(-c3cc(C)cc(C)c3)nc(C)n2)CC12CCS(=O)(=O)CC2.n12cc(nn1)C2 c1(OC)cc(CNC(=O)CN(C(=O)C)C)ccc1OC.C(=O)(C(C)OC1CC1)N N1(C(COCCNC(c2cc(CC)ncn2)=O)=O)CCCC(C)C1C N1(C(C=CCN(C)CC)=O)CC(CNC(=O)COCCF)C(O)C1 c1(C(C2(C(N3CCC(O)(CO)C3)=O)CC2)=O)ccc(F)c(F)c1F c1(C(N2CC(CN(C(=O)CSC(F)F)C)C2)=O)c2ccccc2nn1C N1(C(C(CC)F)=O)CCN(C(=O)CN2Cc3ccccc3C2)CCC1C c1(NC(C2N(c3cc(OC)nc(C)n3)CC(O)C2)=O)ccc(C)c2ncccc12 CC1CC(C(=O)NCC(O)C(C)(C)O)CN(C(c2ccc(C3CC3)o2)=O)C1 C12(COC)CN(C(=O)C3=CCC3)C(CNC(=O)Cc3ccc(F)c(Cl)c3)(C1)C2 c1(C(N2C(CN(C(C(CSC)O)=O)C)CCCC2)=O)ccc2oc(=N)[nH]c2c1 N1(C(COCCCC)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1CCCC n1(CC)ncc(Cl)c1C(N1CCC(C(C)(C)C)(CNC(c2sccc2C)=O)C1)=O C1(CCC)CCC(NCc2csc(CCC)n2)CC1 C1(C(N(C)CC2CCCC2NC(=O)Cc2cn(C)nn2)=O)COC(=O)N1C c1(OCC)ccc(C(=O)NC2CCC(CC(=O)N(C(CO)C(C)C)C)C2)cc1Cl Cc1cc(C#N)ccc1C(N1CC(C(=O)NCC(C)C(C)O)CC12CCC2)=O C1(CNC(CCC(=C)Cl)=O)CCCC2CN(C(=O)COC3CCCCCC3)CC12 Cc1cccc(NC(=O)CCNC(c2c(C)noc2C)C2CC2)n1 c1(C(=O)NC2CCC(CCC(=O)N(CCOC(C)=O)C)C2)cccnc1O N1(C(Cn2cc(C(C)O)nn2)=O)CCN(C(c2cnn(C)c2N)=O)C(CCO)C1 Cc1ccc(Br)c(CC(=O)NCC(F)CNC(c2coc(C(F)F)c2)=O)c1 Cc1ccn2cc(C(N3CCOCC(CNC(=O)C(C)C(C)O)C3)=O)nc2c1 c12nc(C)cc(C)c1C(=O)N2.C1(C(=O)OC)CSCN1C(C(=O)O)C(=O)OC N1(c2nc(SC)c(C)cn2)CC(C2CCCN(C(C3COC(C)C3)=O)C2)C1 CCC(CC)(CCO)NC(C1(CNC(C2CC3CCCC3C2)=O)CC1)=O CC1(NC(c2csc(C(F)F)c2)=O)CCN(C(=O)COC2CCC2)C1 c1(CC(=O)NC(C(=O)NCC=C)C2CC2)ccccc1O CC(C)S(=O)(=O)C(C)C(=O)NCC1CC(O)CN1C(c1ccc(C2CC2)nn1)=O C1(NC(C2(CC=C)CC=CC2)=O)CCCCC1NC(=O)C=C(C)c1cccs1 N#Cc1ccccc1C1(C(=O)NC2CC2NC(=O)C2=COCCC2)CC1 C12(NC(CCCNC(c3ccc(CC)nc3)=O)=O)CCC(C1)OC2C C1(COC)COCCN(C(c2ccccc2)C)C1.c12nccn1CC2 C=CC1OCCCC1C(=O)NC1CC(CCNC(c2cccc(C3CC3)n2)=O)C1 CC1(NC(=O)C=Cc2cccnc2)CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C1 c1(C(N2CC(C(C)NC(CSCCN(CC)CC)=O)C2)=O)ccccc1C C1(NC(C(c2cccnc2)NC(c2ccoc2)=O)=O)CCCN(CC(F)(F)F)C1 C1(NC(C(C)OCCC=C)=O)COCCN(C(c2c(C)coc2C2CC2)=O)C1 CCC(F)(F)CC(=O)N1CC(C)C(C)(CNC(C2CC(=O)N(C3CC3)C2)=O)C1 CC(C)CS(=O)(=O)CC(=O)N1CCCCC1CNC(=O)C=Cc1nccs1 c1(C(=O)NC(CC)CN(C(=O)CNC(=O)OC)C)ccnc2ccsc12 c1(COC)cccc(NCC(=O)NCc2nc(C(=O)O)ccc2OC)c1F Cc1ccccc1C(C)CC(=O)N(CC(C)N(C(=O)Cc1nc[nH]n1)C)C C1(C)(C(N(C(CC)CC)C)=O)CC2CC2C1.C1CC(=O)NCC(=O)O1 C1(CNC(NC(COC)C)=NCC2C3CCCCC23)C2CC3CC(C2)CC1C3 C1(NC(c2ccc(-c3ccco3)o2)=O)CCCCC1NC(=O)C(F)(F)CC1CC1 C1(C(N(C2CCN(CC)C2)C)=O)CCCC1NC(C1(n2nccn2)CC1)=O C(=O)(C(C)C(O)C(C)CC)N(CCC(=O)NC(C)(C)CC1CCC1)CC=C N1(CCOC)CC(C(N2CC(C)(NC(C3CC(C)=NO3)=O)C2)=O)CC1=O C1(N(C(CCC(=O)N(C)C)=O)C)CC2CCC(C1)N2C(=O)CN=S(C)(C)=O Cc1ccc(C=CC(N2CCC(O)(CNC(c3ccc[nH]3)=O)CC2)=O)cc1Cl C1(C(=O)NCC(CC=C)NC(C)=O)C2CN(C(c3ccccc3F)=O)CC12 CC1C(C(=O)N(CCN=[N+]=[N-])C)CCN1C(=O)CCc1cn[nH]c1 Cc1ccc(C)c(C(=O)NC2CN(C(c3ccc(C(N)=O)[nH]3)=O)CCC2F)c1 C1(C)(C(=O)NCCC2CCCC(C)C2)CCCN(C(=O)Cc2n[nH]c(=N)s2)C1 CC1CCC(n2cc(C(N3CCC(O)(C(N(C)C)=O)C3)=O)nn2)CC1 N1(C(C2C(CNC(C3(CCCC)CC3)=O)CCC2)=O)CC2(C1)CN(C)C2 C1(NC(CC2CCN(C)C2)=O)CCOCC1C(=O)NCCS.N1(C2CC2)CCCC1 N1(C(=O)COCCF)CCN(C(=O)COCC2CCCCO2)C(CC(F)F)C1 c1(C(N)=O)cccc(C(C2CC2)C(C2CC2)O)c1.CC12CCN1NC(=O)C2 N1(C(C2(C#C)CN(C(CCCOCC)=O)C2)=O)CCN(CC)C(C)C1 C1(C(C)(C)C)CCCCC1C(=O)NCC1CC(CNC(=O)Cc2csc(=N)[nH]2)C1 N1(C(C(CC=CC)CC)=O)CCC(C)(C)C(C(N2CCOC(CC)C2)=O)C1 Cc1cnc2n1C(C(=O)NC1CN(C(C3(C#N)CC3)=O)CCC1(C)C)CCC2 CC1(C2(C(=O)NC3CCC3c3cn(CC(N)=O)nn3)CC2)CCCO1 c1(N(C(c2ccsc2NC(=O)OC(C)(C)C)C(=O)NC(C)C)C)cccc(Cl)c1 C1(C2CN(C(=O)CCCC3OCCO3)C2)(NC(CC2N(C)CCOC2)=O)CC1 C1(CNC(c2nnnn2C2COC2)(CC)C2CCC2)CC2C(C1)C2(F)F N1(C(CC=CC=C)=O)CCCN(C(=O)CC2CCCCC23CC3)C(CO)C1 C#CCCCCCCC(=O)NC1CCCC1C(=O)NC(CC#C)CC#C c1(C(=O)NC2CC(C(N3CCC(Br)C3)=O)C2)ccccc1F c1(C(N2CC(F)CC(NC(C(CC)O)=O)C2)=O)noc2c1CC(F)(F)CC2 c1(C(=O)NCCC2OCC(C)(C)C2)csc2cc(Br)cnc12 Cc1c[nH]cc(-c2nc(-c3ccncc3)nn2Cc2ccc(C(F)F)cc2)c1=O O=C(C#CC1CCC1)N1CCN(C(=O)C(O)(C2CCC2)C2CCC2)CC1CO C1(CC)C(C(=O)NCCCN(C)CCOC)CCN1C(c1cc(C(C)=O)c[nH]1)=O CCS(=O)(=O)CC(=O)N(C1CCC(NC(c2cnc(C3CCOC3)s2)=O)CC1)C n1(CC)nc(C(F)(F)F)cc1C(=O)NCCCNC(C1CCC1n1ccnc1)=O c1(NCC2N(C(c3ccc(C(C)O)cc3)=O)CCC2)cc(=O)n(C)c(=O)n1C C(=O)(C(C)CSCCCCC)O.C1(SCC)CC1 N1(C(c2ncc(C)cc2C)=O)CCC2(CC1)OCCC2NC(=O)C1=CCCCO1 CCCCC(CNC(C1(CO)CC(C)(C)C1)=O)NC(C1CC2CCC2C1)=O C(=O)(C(C)CCCC)N1CCC(C2N(C(CC=C=C)=O)CCC2)CC1.C1CC1 C(CCCCNC(C1(CF)CC1)=O)N(C)C(C1CC1c1ccsc1)=O N1(C(c2cc(C)[nH]n2)=O)CCOCCC1C1CC1.C(C(=O)NCC1CC1)(C1CCC1)OC C1(CC=C)(NC(=O)C(C)c2cccs2)CN(C(c2cn(CCOC)nn2)=O)C1 C1(=CC(=O)NC2CCN(C(C(C)c3ccsc3)=O)C2)C2CC3CC(C2)CC1C3 CC1=NNC(=O)C1CC(N1CCC(CNC(c2[nH]c(C)nc2C)=O)C1)=O C1(C(=O)NC2C(C)CN(C(=O)C=C3CCC3)C2)COc2cc(Cl)ccc2C1 CC1CCC(NC(=O)CCn2ccnc2)CN1C(C1COC(C)(C)CO1)=O c1(C(=O)NCc2ccc(C(=O)NCCCOC(C)C)o2)ccc2[nH]ccc2n1 C(CC(O)C(=O)N1CC(c2nc(C3CC3)no2)C1)CC(=O)NC1CCOCC1 Cc1nc(CO)ncc1C(N1CCCCC(NC(=O)CCC2CC2(C)C)C1)=O c1(NC2CC3CN(C(=O)OC(C)(C)C)C2C3)ccnc2ncnn12 CC(C)CC(CNC(=O)CC1CC(C)(C)CO1)NC(c1cccc(Cl)c1)=O c1(CNC(=O)COC2COC2)cccc(-c2cncnc2)c1 C#CC(CNC(=O)C(CNC(=O)C(C)(C1CCCC1)OC)N(C)C)CC n1(C(CC)C(=O)NCC2(NC(c3ncn(CC)n3)=O)CC2)cnc(C#N)n1 c1(OC)ccc(OC(F)F)c2cc(C(=O)NCC(C)(C)n3ccnc3)[nH]c12 N1(CC(N2CCC(C(C)NC(C3(F)CCOC3)=O)C2)=O)CCCCCC1=O Nc1nc(C(=O)NCC2CC2CNC(c2cnc(-c3cccs3)o2)=O)ccc1O C12(C(=O)NCC3N(C(c4ccc(Cl)o4)=O)CC(F)C3)CCCN1S(=O)(=O)CC2 C1(CC)CCN(C(c2ccn(CC)c2C)=O)C(C(=O)N(CCN(C)C)CC)C1 C=CC(C)(CC)C(=O)NC1CCC(NC(=O)COC2(C)CCCC2)C1 c1(-c2cn(CC(=O)N(C3CCCCC3)CC#C)nn2)ccncc1C#N C1(OC)CC(NC(c2ccc(F)cc2Cl)=O)CN(C(=O)Cc2ccc(O)nc2)C1 C1(C(N(C2CN(C(c3ccc(N4CCC4)nc3)=O)C2)C)=O)CCC(F)(F)C1 N1(C(COC(CC)C)=O)CCC(NC(c2ccc(C)c(N)c2)=O)C2(CCC2)C1 c1(N2CCN(CCCNC(CC(CC)OC)=O)CC2)cc(=O)n2oc(C)cc2n1 c1(NC(c2nc(-c3ccc(C)c(C)c3)sc2C)=O)cc([N+](=O)[O-])ccc1Br N1(C(CSCCCC)=O)CCC(NC(c2ccc(C(F)(F)F)c(Cl)c2)=O)CC1C CC1(C)CCCC(C)(C)C1C(N1CCN(C(=O)C(F)F)C(C2CC2)C1)=O Cn1ncc2c1CCCC2Nc1cc(Cl)c(S(=O)(=O)NC2(CF)CCC2)c(Cl)c1 CC(C)C(O)CC(=O)NCC1(F)CCC(CNC(c2ccc(C(C)(C)C)o2)=O)C1 N=c1cc(-c2cn(CCCC(=O)NC3C(O)C4CCOC34)nn2)cc[nH]1 C(=O)(C(CC(C)C)OC)NCC(=O)N(CC(F)F)C(c1ccccc1)C C1(NC(Cc2n(C)nnc2)=O)CCC2CN(C(=O)Cc3ccccc3O)CC2C1 Cc1nc([N+](=O)[O-])cn1CCC(=O)NC(C)CNC(c1n[nH]cc1C(C)(C)C)=O c1(NC(C2C(NC(CCOC(C)=O)=O)CCC2)=O)cc(Cl)ccc1C Cc1nc(C(=O)NCC2(C)CCN(C(=O)CC3CCCO3)C2)c(C)s1 N1(C(C2(SC)CCC2)=O)CC2C(CN(C(=O)CC3CCOC3)C)C2C1 C1(CNC(C2CCC(C)C(C)C2)=O)CC2CCC(C1)N2C(c1nccnc1Cl)=O c1(-c2cncc(C(N3CC(C(C)(C)O)C3)=O)n2)ccc([N+](=O)[O-])cc1F C#CC1(C(=O)Nc2conc2C)CN(C(=O)CN2C(=O)CNC2=O)C1 CC12CCC(C(=O)NC3COCCC3NC(c3ccncc3Cl)=O)(C1)OC2 C1(CNC(CCN(CCC(C)(C)C)C)=O)COCCN1C(=O)Cc1ccnn1C C=CCCCCCCCC(=O)NCC1(CNC(C2CCOC2)=O)CCC1 c1(C(=O)NC(C)CN(C(=O)CCc2cscn2)C)nn[nH]c1C(F)(F)F Cc1nc(C(=O)NCC(C)N(C)C(c2ccn(C3CCCC3)n2)=O)c(C)o1 Cc1nc2c(N3CCC(NC(c4cc(F)c(F)c(O)c4F)=O)C3)ncnc2[nH]1 Cc1scc(C(=O)NC2CCC(CCNC(=O)C(F)(F)C3CC3)C2)c1C CC(C)CCCCC(=O)NC1CCN(C(c2cnn(CCO)c2)=O)C12CCC2 C12(CNC(Cc3c(C)non3)=O)CCC1CCN2C(c1cnn(C(C)C)c1N)=O C(N=c1cc(C2CC2)n(C)[nH]1)(c1c(OC)csn1)c1nnnn1CC(F)F c1(C(C(=O)NC(CC(C)NC(c2n(CC)ccn2)=O)C)(F)F)ccc(F)cn1 N1(C(Cn2c(C)ncc2)=O)CC(CO)C2(C1)CN(C(C1CCCCC(=O)N1)=O)C2 c1(C(=O)NCC2=CCN(C(C)C(N)=O)CC2)cc2cc(Cl)ncc2[nH]1 C1(NC(C=C(C)Cl)=O)CC2(C1)CC(CNC(=O)C=C(C)CCc1ccccc1)C2 CCC(CCC(=O)NC(C)(CO)C(=O)N1CC(CC(F)(F)F)C1)OC O=C(CCCC(F)(F)CO)NCC1CC2CCCC2N1C(=O)Cn1cnnc1O N1(C(C(COCC)C)=O)CC2(CC)CC1(CNC(=O)C(c1ccccc1)C)C2 C(=O)(CC(C)CC(=O)NC1CCC1CC(=O)NCCC1(CO)CCN(C)C1)OC CC1C(C(=O)NCC2(CN(C)C)CC2)CCCN1C(c1ccncn1)=O c1(C(=O)NCCN(C)C(c2cc(-n3cnnc3)ccn2)=O)cc(S(N)(=O)=O)cs1 c1(C(=O)Nc2scc(C(C)(C)C)n2)cccc2occc12 C1(CC(=O)NCC(CNC(C(C)n2cccc2)=O)O)CC(C)(C)C(=O)N1 C1(C)(C(=O)NCC(COC)NC(=O)CCCCNC(C)=O)CCC(=O)NC1 C1(F)(C(=O)NC(c2cnc[nH]2)C)CCCN(C(=O)C(N2CCCCC2=O)C)C1 CCCCC(F)(F)C(=O)N1CCN(C(=O)Cc2cc(C3CC3)on2)C(C(C)C)C1 N1(C(C(C)OCC=C)=O)CCC(C(N2CC(O)C2)=O)C(c2ccccc2)C1 c1(OC)ccc2occ(C(N3CCOC(Cc4ccccc4)C3)=O)c2c1 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CC(NC(=O)CCc1cccn1C)C2 N1(CCN(C(=O)NCCNC(c2ccc(C)cc2)=O)C)CCC2CCC(O)C1C2 c1(C(=O)NC2C3CN(C(=O)CC4CCC(F)(F)C4)CC23)cc(F)cc2c1CCC2 c1(CCN(c2nc(C(c3sccc3Br)C3CC3)no2)C)ccc(F)cc1 c1(C(=O)NCCC2CCCN(C(CN(CCOC)C)=O)C2)cccc(CO)c1C C(=O)(C(F)CC(C)(C)NC(=O)C=C1CCCCC1)NC(C)CN(C)C c1(SC)cc(C)ccc1C(N1CCC(C)(NC(C2CC(=O)C2C)=O)C1)=O c1(C(=O)NCC2CC(C(=O)NC(C=C)C3CC3)C2)cc(Cl)ccc1Cl C1(NC(C(CC=C)(C)N(C)C)=O)CC2CC1CN(C(=O)C=C(C)c1ccccc1)C2 C1(C(=O)NC)CCCOCC1.c1(C(N)=O)ccc(C(N2CCC2CSC(F)F)=O)o1 C1(CNC(CCOCC(C)C)=O)CC(C(=O)NCC(C)CN(C)C)=NO1 c1(-c2cccc(OC(c3cscc3OC)C(=O)OC)n2)ccc(O)c(C(N)=O)c1 c1(C2CCN(C(=O)Oc3ccccc3)C2)cccc2ccccc12 Cn1cnc2c(N3CC(CNC(=O)CC4OCCC4(C)C)C3)nc(Cl)nc12 C1(C(=O)NCCCCCCN(C(=O)Cc2csnn2)C)(CC)CCCCO1 C1(CN(C(=O)CCc2ccc(=N)[nH]c2)C)CN(C(c2ccncc2Br)=O)CCO1 c1(C(C(=O)NCC2COC(C)(C)O2)N2CCCC2)cc(Br)cc(Br)c1 Cc1nc2n(n1)CC(C(=O)N(CC(O)CNC(C1(S(N)(=O)=O)CCC1)=O)C)CC2 c1(OC)ccc(CN2CCN(C(=O)NCc3cnc(F)c(C)c3)CC2)cc1OC c1(C(=O)NC2CC2)cccc(OC)c1.C12CC1C(=O)NCCN(CC#C)C2=O N1(C(c2cc(C)ncc2Br)=O)CCC2(CC1)COCC(CO)O2 C1(CNC(CCc2n(C)ccn2)=O)CCCCCN1C(c1cc(N)ccc1Cl)=O c1(C(N2CC(O)CC(NC(c3nc(CC)oc3)=O)C2)=O)cc2ccccc2n1C C1(C2CC2)(NC(c2nc(C(N)=O)sc2)=O)CCN(C(C2CCCC(F)C2)=O)C1 C1(C(=O)NC2COCC2CO)CCCCN1C(c1cccs1)=O C(CC(C)C(=O)NC(C)(CNC(=O)Cc1ccccc1)C1CC1)=CC Cc1ccc(C)c(CC(N2CC(CNC(=O)C(C)N3CC(C)C3)C(C)(C)C2)=O)c1 c1(C(C(N2CC(CCNC(c3[nH]ccc3C)=O)(OC)C2)=O)=O)ccc(C)cc1 CC1(NC(C2CCNC(=O)C2)=O)CCC(NC(c2cc(F)cnc2O)=O)CC1 c1(C(=O)NCC2CN(C(C3(SCC)CC3)=O)C2)cc(F)cc(F)c1N N1(C(Cc2c(C(C)C)con2)=O)CCC(NC(=O)CCC(=O)N(C)C)C(O)C1 C1(NC(C2(CCCC)CC2)=O)CCCCC1NC(=O)CCN(C(C)CCC)C1CC1 C(=O)(C(=O)C(C)C)N1CC(CC(=O)NCCC=CCCC)C1 c1(C(=O)NC2CN(C(CC=CC=C)=O)CC2C)ccn2[nH]c(=N)nc2c1 c1(NCC(CCCC)NC(c2cn[nH]c2)=O)nccc(C(N)=O)c1[N+](=O)[O-] n1(C2CN(C(C(=O)N(C3COC3)Cc3c(CC)cno3)=O)C2)nc(C)cc1C Cc1nn(CC(C)C)c(C)c1CN(C1CCCC(C)(C)C1)CCOCCO C1(C(N2CC(C(C)NC(C3C(CC)CCCC3)=O)C2)=O)CC(=O)NC1(C)C Cc1[nH]nc(C(=O)NC2CC(C)CN(C(=O)C(=O)NCC(F)F)C2)c1[N+](=O)[O-] CC1CCCN(C(=O)CCn2cncn2)C1CCNC(=O)CCN1CCCC1=O c1(N2CC3N(C(C4CC(=O)NCC4)=O)C(CC3)C2)[nH]cnc2nc(Br)cc1-2 CC12CN(C(C34CC(CN3C(C3CCC3)=O)C4)=O)CC1(CO)C2 N1(C(C2C(C(=C)C)OCC2)=O)Cc2ccc(CNC(=O)C(F)C3CCC3)cc2C1 c1(OC)cccc(I)c1NC(C1CN(Cc2ccc(O)c(O)c2)CCS1)=O C(C(=O)N(C(C)CNC(=O)CN1CC2CC2C1)C)(C(C)C)OCCOCC C1(CNC(c2ncc[nH]c2=O)=O)CN(C(C2CCCC3(CC3)C2)=O)CC12CCC2 Cc1c(NCCC(=O)N2CCC2C(=O)NC2COC2)cnn1-c1ccccc1 N1(c2c(C)c(N3CCC(=O)C4(CCC4)C3)ncn2)CCN2C3=NC=CC(C3)C2C1 CC1CN(C(=O)C(C2(O)CCCC2)F)CC(C)N1C(c1nnc(S)n1C)=O C1(N(S(Cc2nc(C)sc2)(=O)=O)C)CCC(C(F)(F)F)CC1 C1(NC(C(CC)=CC)=O)Cc2ccccc2C1NC(c1ccc(Cl)nc1O)=O N1(C(C(C)CC(N)=O)=O)CC(CNC(=O)C=Cc2ccc(F)cc2)CC12CCC2 C1(C(=O)NC2CC2c2ccccc2)C2CCC(C2)N1Cc1cccnc1O C1(CC=C)(NC(=O)C(C)(C2CCC2)NC(c2occc2C)=O)CCCC1 c1(OC)ccc(C(N2CCC(O)(CCNC(C3(CO)CCCO3)=O)C2)=O)cc1C C(CC(CO)N=c1ccn2ncc(C(=O)NC(N3CCNC4CNCC34)=O)c2[nH]1)=CC C1(Nc2ccc(N3CC(OCC)C3)c(F)c2)CNC2(CCCOC2)C1 c1(C(=O)OCC)cc(C)ccc1NC(=O)C(=O)N(C1CCS(=O)CC1)C c1(C(=O)NC(C(C)NC(=O)CC2CCCC2)CO)cc[n+]([O-])cc1 c1(C(N2CC=CC(C(=O)N(CC3CC3)CC3CC3)C2)=O)ccc(O)cc1F C(=O)(C(C(C)(C)C)N1CCOC1=O)NCCCNC(c1ccc(SCC)cc1)=O C1(C(=O)NCCC(=O)NC)CC2(CC(NC(C3CC3(Cl)Cl)=O)C2)C1 c1(CNCC(N)=O)ccc(C(c2nnnn2C2CC2)OC)cc1 c1(C(N(C2CCN(C(c3snc(O)c3Cl)=O)C2)C)=O)n[nH]c2c1CS(=O)(=O)CC2 c1(C(=O)NC(C)C(=O)NC2(C)CC(NC(=O)C(F)=C3CCCC3)C2)ccccn1 N1(C(c2cn(C)cn2)C(=O)Nc2c(C)c(Cl)ccc2)CC(=O)NCC(C)(C)C1 C1(CC(=O)NC(CC(=O)NCC2(CC)CC2)C2CC2)CCC(C)(C)O1 CN1CCCCC(C(N2CCOC(C(F)(F)F)(C3CCC3)C2)=O)C1=O C=CC1(C(=O)NC2C3CCCOC23)CCN(C(c2cncc(C#N)c2)=O)CC1 c1(C(N2CC(C)(C)C(NC(C3(C)CCC(F)(F)C3)=O)C2)=O)c(N)cc(Cl)cc1F CC1CC(=O)CCC1C(N1CCC(NC(=O)C2=COCCO2)C(F)C1)=O c1(OC)ccc(OCC(=O)NC2CCCCC2NC(c2nn[nH]c2Cl)=O)cc1 c1(C(=O)NCC2C(CNC(C(N)=O)=O)C2)occc1F CC(C)CC(C(=O)N1CCC1C(C)(C)O)ONC(=O)C1CC1 N1(c2cc(COC)ncn2)CCC(NC(c2ncc[nH]2)=O)C2(CCC2)C1 c1(C(=O)NC(CCNC(C(C#C)(C)C)=O)C)coc2c1CS(=O)(=O)C2 Cc1cc(C(=O)NC2CCN(C(c3ccc4nc[nH]c4c3)=O)CC2)c(C)nc1C Cc1cc(C)c(NC(=O)C(=O)NC(=O)CCC2CCC(NC(C)(C)C)O2)c(Cl)c1 C1(C(F)(F)F)(C(=O)NC(C)CCNC(=O)C(c2ccnn2C)C)CC=CCO1 C12(C(N3CC(O)(CNC(CS(C)(=O)=O)=O)C3)=O)CC=CC(C1)OC2 N1(C(C(NOC)=O)=O)CCC(C)C(NC(C2CC3CCC2C3)=O)C1C c1(C(=O)NCC2CN(C(C3C(C)OCCC3)=O)C2)c(N)cccc1[N+](=O)[O-] c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cc(C)c(Cl)s2)=O)C(CO)C1)=O N(C)(C1c2ccccc2CCC1C)C(=O)NCC(C)SC C1(CNC(=O)CCC2CCOCC2)CCN(C(C2CCOC(=O)CC2)=O)C12CC2 c1(CCC)ccc(NC(=O)C(C2CC2)NC(C2CCCOC2)=O)cc1 c1(OC)ncc(Cl)c(C)c1C(N1CCOCC(CNC(C2CCCN2C)=O)C1)=O C(=O)(N=c1cc2n([nH]1)CCCC2)C1CCN(C(C2C(C(=O)OC)C=C2)=O)C12CC2 C1(C(N(CC)Cc2cn[nH]c2)=O)C=CCCN1C(C1CCS1(=O)=O)=O C(=O)(C(C)(F)C(C)(C)F)N(CC(CNC(c1c(CC)n(C)nn1)=O)(C)C)C c1(C(N(C)CC2CCCN2C(C2CC3CCC2O3)=O)=O)ccnc2c1CCO2 Nc1nccnc1C(=O)NCCC1(O)CN(C(=O)C(F)CC2CCCC2)C1 C1(CNC(c2c(NC)snc2C)=O)CCN(C(c2scc(C)c2Cl)=O)C12CC2 C#Cc1ccc(C(N2CCC(O)(C(C)NC(=O)COCCN(C)C)C2)=O)nc1 C1(CNC(c2ccc(C(N)=O)[nH]2)=O)CN(C(=O)C(F)OC(F)(F)F)CCO1 c1(NC(C2CCN(C(c3ccno3)=O)C2)=O)cc(F)c(Br)cc1F C(=O)(C#CC1CCOCC1)NC(CN(C(c1scc(OC)c1OC)=O)CC)C C(=O)(C(C)(C)C(C)(C)O)N1CC(O)CC(NC(CCCONC(=O)OCC)=O)C1 N1(C(C2(C)CNC(=O)N2)=O)CC2(CCOCC2)CC1CNC(=O)CC1CCCO1 C(CN=c1[nH]cnc(C)c1F)(CC(C)C)NC(c1c(C)n[nH]c1C)=O c1(N(C)C(C2CC2c2ccccc2N)=O)ccc(F)c(C(F)(F)F)c1Cl Cc1cc(CC(=O)NCC2CN(C(=O)CCC3CC3(F)F)CCO2)cc(C)c1 C1(NC(CC(C(C)C)OCC)=O)CC2CCC(C1)N2C(c1coc(C(N)=O)c1)=O c1(C(=O)NC2(CCOC)CCN(C(=O)CCC3CC3(C)C)C2)ccc(Cl)cc1C Cc1nn(C)c(C)c1CCC(N1CCC(C(C)NC(c2n[nH]c(=N)s2)=O)C1)=O c1(CNC(C2CCSC2)C)[nH]c(=NCCc2cnc(C3CC3)nc2)nc2scnc12 CCC(CC)(CO)C(=O)NC1(CNC(c2cnc(C3CC3)o2)=O)CC1 O(NC(=O)C(F)CC(C)(C)NC(C1CC1C1CCC1)=O)C1CCN(C)C1 c1(OC(C)C)cccc(C(=O)NCC(CNC(c2cc(N)ccn2)=O)CO)c1F c1(CC(=O)NC(C2CCN(C(Cn3c(C)cnc3)=O)C2)C)n[nH]c2ccccc12 C1(C(=O)NCC(C)CC2CC2)CCC(C)CN1C(c1ccc(CN(C)C)nc1)=O N1(C(C(=O)NCCOCC)C2CC2(C)C)CC2CN(C)CC(C1)O2 N1(C(CSC(C)(C)C)=O)CC(CO)C2(C1)CN(C(=O)CNS(C)(=O)=O)C2 Cc1cc(CCC(=O)NC2CC(NC(C34CCC(C3)C4)=O)C(O)C2)cc(C)c1 C1(NC(C(CC)n2cncn2)=O)CCC2CN(C(=O)Cc3csnn3)CCC2C1 n1(CCC(=O)OCC)nc(-c2ccc(C)cc2)nc1Cc1cccc(C)c1 C(=O)(C1=CC2CCC=CCCC12)NC(CNC(c1c(C)n2c(s1)ncc2)=O)(C)C C1(NC(C(CC#C)C)=O)CN(C(C2CN(C)CC(C)O2)=O)CC1(C)C c1(C(=O)NCCC(C)(C)NC(=O)C(C)(C)c2cscn2)cc(Cl)ccn1 C(=O)(CCC(C)(C)C#N)N(CC(C)C(=O)N(C)CC1CCCC2CC12)C C1(NC(C(C)=C2CCC2)=O)CC12CCN(C(=O)C1=CC3C=CC1C3)CC2 c1(C(=O)NC(CN(C(=O)C2=NNC(=O)CC2)C)(C)C)ccc2ncccc2c1F C1(CNC(C2CC=CCC2)=O)CCC(NC(=O)C(C2CC2)C2CC2)CC1 C(=O)(C(CC1CCCO1)C(C)C)NCCCCC1CN(C(c2cc(C)c(Cl)s2)=O)C1 C1(CCN)CN(CC2CCCCCCC2)CC12CC2 C1(n2c(C)cnc2)CCN(C(=O)C(n2ccc(C(F)(F)F)n2)C)CC1 C1(CC(=O)NCC2C3CN(C(=O)Cc4sccc4Cl)CC23)CCCOCC1 c1(N(C)CC2CN(C(C(COC)O)=O)C2)ncc(C(F)(F)F)cc1Cl Cc1ccn2ncc(C(=O)N(C3CCC(NC(C4(CCF)CCC4)=O)C3)C)c2c1 C1(NC(CCOCCCOC)=O)CC(C)(NC(c2ccc(C(C)=O)o2)=O)C1 C1(CBr)CCCN2N(Cc3ccc(F)cc3)C1CCCC(F)C2 CCC(F)(F)C(=O)NC1CN(C(c2cc(C#N)on2)=O)CC1OC C(C(CC)CCO)NCc1nnnn1CCC(CCOC)SC.c1(CC)noc(C)n1 C(CN=c1[nH]c(=NCC23COC(C2)C3)[nH]c2cccc(F)c12)C1C(O)COC1 N1(C(c2ccc(N(C)C)nn2)=O)CC2(CCN2C(c2ccc(CCO)cc2)=O)C1 C1(C(N2CCN(CCCNC(C3(C#N)CC3(C)C)=O)CC2)=O)(CC)CC=CCC1 c1(CN(C(c2c(C)noc2)C(=O)NCC(C)C)C2CC2)cccc(CO)c1 C=CC(C)(O)C(=O)NC(C)CCNC(=O)CC1COCC1(C)C C1(CC(N2C(CCNC(c3c(CC)occ3)=O)CCC2)=O)CCC(C#N)C1 Cc1nc(C)c(CC(N2CCC(NC(C3CC(O)C3)=O)CC2)=O)c(O)n1 CCC(C)C(CO)NC(C1C=CCCN1C(=O)C(C)N(C)C(C)=O)=O C1(NC(=O)C2=CCSC2)CCN(C(=O)C=C(Cl)Cl)CC1F C=CCCCCCCC(=O)NCC=C1CCN(C(c2ccc(Cl)nc2N)=O)CC1 c1(NCCc2c(Cl)ccc(O)c2)ccnc2ccc(I)cc12 C1(C(N)=O)CCCC(C(=O)NCCC2(CNC(c3csnc3Cl)=O)CC2)C1 Cc1noc2cc(C3CC3C(=O)Nc3ccc(F)c(O)c3)ccc12.C1CSCC1 c1(C(=O)NC2C=CCN(C(Cc3c(C)cccc3)=O)C2)cn2cccnc2n1 C12CCN(CC1)C(=O)C2.C1(NC(=O)CC2CC(CCF)C2)(CF)CC(F)(F)C1 Cc1ccc(-n2cc(C(=O)NC3CCN(C(=O)C(F)F)C3C)c(C)n2)cc1 c1(C(=O)NC(C2CCCCC2)C(=O)NC(CSC)C)ccc2ccoc2c1 c1(CC(=O)NC2(CCNC(C3CC3Cl)=O)CCCC2)ccncc1Cl CC(C)(CC(F)(F)F)C(=O)NCC1CC(F)CN1C(C1Cc2nccnc2C1)=O N1(C(C2C(CNC(C(c3ccnn3C)C)=O)CCO2)=O)CC2(COC(=O)N2C)C1 c1(CCNC(C(C2CCCOC2)N(C)C)=O)ncccc1Cl C12(NC(C=C(CC)CC)=O)CCCCCC1N(C(c1cnc(F)c(Cl)c1)=O)CC2 C(=O)(CC(C)(C)C(F)F)NCC(C)(Cn1cccn1)NC(CC(C)C1CC1)=O N1(C(C(c2ccccc2F)C)=O)CCN(C(c2cc(Cl)ccn2)=O)CCC1C C1(F)(C(=O)NCC2CCC(F)(F)C2)CCCN(C(C2(Cl)CC2(F)F)=O)C1 c1(C(=O)NC2CN(C(c3ccc(C4CC4)nc3)=O)C3CC23)cccc(F)c1Cl c1(C(C)C)nn(C)c(C(N2CCC3CC2CO3)=O)c1Br.N12CCCC1SCC2=O C(=O)(CCCCC(C)C)N(CCCC(N1CC(C)(CC)C1)=O)C C1(OC)CCC2(C(=O)NC(C)C(C)(C)NC(c3cnc(O)c(C)c3)=O)CCC12 c1(C(=O)NCC(C)NC(C2(C)COCCO2)=O)cnc(C2CC2)nc1O C1(C(C)C)CN(C(C2COCCN2C)=O)CCN1C(c1csc(C(F)F)n1)=O C1(C(N2C(CCNC(c3[nH]cc(CC)c3)=O)COCC2)=O)CCn2nncc2C1 c1(C(=O)NC2CC(CNC(C34CCCCC3C4)=O)C2)coc(=O)c2ccccc12 c1(C(=O)NCC(=C2CN(c3cc(Cl)c(O)nn3)C2)F)cc2ccccc2[nH]1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)C(C)C2(O)CCC2)CCC1C C(CCCC(=O)NCC(C)(C(C)C)NC(C1CCN(CC(F)(F)F)CC1)=O)OC C1(NC(C2CCSCC2)=O)CC2CN(C(=O)CCCCCF)CC2C1 C=CCCC(CC(C)C)C(=O)NC1CC2(C1)CC(NC(=O)C(F)C(C)C)C2 C1(CC)CN(C(c2cnc(CO)nc2C)=O)CCN1C(=O)C=C(C)c1ccsc1 CC1(C)CCCC(C(=O)NCC(O)CC(=O)NCC2CCOCC2)C1 C(C(CC(C)C)NC(c1cc(-c2ccc(O)cc2)on1)=O)NC(C(C)=CC)=O c1(NC(C2CN(C3CN(C(C(C)(F)F)=O)C3)C(=O)C2)=O)cc2ncccc2[nH]1 c1(C(=O)NC2CCC(NC(=O)C(c3ccccc3)F)C2)ccc2c(n1)CCOC2 Cc1ccc(C(N2CCC(O)(CNC(c3cnn[nH]3)=O)CC2)=O)c(N)c1Br c1(C(N(CC(CNC(c2n(CC)cnn2)=O)O)C)=O)cccc2c1OCCC2 c1(NC(=O)NCC(CCC(=O)OCC)(F)F)cncc2nccnc12 S(=O)(=O)(c1ccc(C)c(C)c1)NCCC(=O)NC1C(CNC(C(C=C)(C)CC)=O)C1 c1(OC)ccc(OCCCNC(c2nc(-c3cccs3)cs2)=O)cn1 c1(C2C(C(=O)NC3CC(NC(CCc4cc(OC)no4)=O)C3)C2)ccc(Br)cc1 C(CN=c1[nH]cncc1I)OCCN(C(=O)CC(C)(F)F)C CC1CCN(C(c2ccnn2CCF)=O)CCN1C(C1OCC1(C)C)=O C(CCCCC(=O)NCCCCNC(COC)=O)NC(c1cc(C)cc(O)n1)=O C1C(C)(OC)C(=O)N1.c1(CCCNC(C2CN(C(=O)NC)C2)=O)nocc1C c1(CC)ccc(C(C)=CC(=O)N(C)CC2CCCN2C(C2CC2F)=O)cc1 CC(C)C(C(=O)N1CCC(CNC(c2cnn(C(C)C)n2)=O)CC1)n1cnnn1 C1(C(N2CC(CC(COC)(C)C)C2)=O)CCc2ccccc2O1.C12CC1C(=O)N2 C1(CNC(C2C(C)=CCS2)=O)CC(C)CN(C(C2(O)CCSC2)=O)C1 C(=O)(C(F)(F)CC(C)C)NC(CC=C)CNC(=O)Cc1c[nH]ccc1=O C1(C(N2C(C(=O)OC)CC2)=O)CCCCC1(C)NC(=O)Cc1cccnc1F CCC(CC)CCC(=O)NC1CN(C(=O)C(c2ccc(F)cc2)=O)CCC1C C1(CNC(C2C(C)C2)=O)CN(C(=O)CCCC2CCCC2)CC12CCC2 N#Cc1ccc(CNC(c2cccc(-c3ccno3)c2)=O)cc1 Cn1nnnc1C(c1conc1C(F)(F)F)NC(C)(C)CCF S(=O)(=O)(CC(C1CC1)OCC1CC1)NS(=O)(=O)Cc1ccccc1 c1(C(N2CC=CC(NC(CCCNC(N)=O)=O)C2)=O)ccc(CO)cc1F C1(CNC(Cc2nc(C)c(C)[nH]2)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C12CC2 C1(NC(C2C(CC(C)(C)C)C2)=O)C2CC1CN(C(=O)OC(C)(C)C)C2 N1(C(C(C)N2CCC2)=O)C2CCC1CN(C(C1(C)CCCNS1(=O)=O)=O)C2 C1(O)(CNC(C2CCC(CC(C)C)CC2)=O)CCN(C(c2ccsc2Cl)=O)CC1 C(C(CNC(=O)C(F)CC1CCOC1)S(C)(=O)=O)Nc1nccc(C(=O)OC)n1 Cc1nn(C)c2ncc(C(=O)N(CCCN(C)C(C3CCC3F)=O)C)cc12 C1(CNC(Cc2ccc(C)s2)=O)CC(F)(F)CN1C(=O)CCOC1CCC1 c1(C(=O)NC2CCN(C(Cc3ncc(C)s3)=O)C2C)cc2n(n1)CCCC2 Cc1ccccc1C(=O)NC1(CF)CCN(C(=O)CCCn2cncn2)C1 N1(C(CC(=O)OC)=O)CCCOC(CCNC(c2cnoc2-c2ccoc2)=O)C1 C12(C(=O)NCc3ccc(C)nc3)CCN(C(c3c[nH]cc3C)=O)CC1C2 N1(C(CCOC(C)=O)=O)CCC2(C1)CN(C(=O)Cc1ccnc(F)c1F)CC(C)O2 N1(C(CCCN(C)CC2CCC2)=O)CCCC(C(=O)NC2CCCC(=O)N2)C1 C12CC3CN(CC13)C(=O)c1nnsc1C(=O)N2.c1(CC)ccc(Cl)nn1 N1(C(C(CC)C)=O)CCC(NC(=O)Cc2ccsn2)C1(C)C C(=O)(C1=NNC(=O)CC1)N1C(CN(C(=O)CCCCn2ccnn2)C)CCC1 C1(C(N)=O)C2CNCC12.C1(c2cccs2)(NC(c2ccc(N)cc2)=O)CCOCC1 c1(C(=O)NCC(CCOC)NC(c2ncn(CC)n2)=O)cc(C(C)C)ccc1F c1(CCC)cc(C(=O)NCc2ncoc2CCNC(=O)Cc2cscn2)sc1C Cc1csc(=NCC(=O)NCC2CC(O)(CNC(c3c[nH]nc3Br)=O)C2)[nH]1 CCC(C(=O)NC1CC(C)(NC(=O)Cc2csc(C(C)OC)n2)C1)C(C)O N1(C(c2n[nH]c(C)c2F)=O)CC2(CCN(C(=O)CCc3ccccc3Cl)C2)C1 Cc1ccc2nc(SCC(=O)OC(c3cccs3)CN3CCOCC3)[nH]c2c1 N1(C(C2(F)CCCN(C(Cn3ncc(C)c3)=O)C2)=O)CCCC2(CC1)CC2 c1(OC(=O)OC(C)(C)C)cccc(C(N2CC(C3C(C(F)(F)F)C3(F)F)C2)=O)c1F c1(C(=O)NC2CC(NC(Cc3c(C)noc3Cl)=O)C2)cc(C)c2[nH]cnc2c1 C1(CC=C)CCN(C(C2CC(CCNC(c3cncn3C)=O)C2)=O)C1 C1(CCC)CN(C(C2(CC(C)C)CC2)=O)CCN1C(C1OC2CCC1C2)=O CCCC(C(=O)N1CC(N(CC)CC)C1)NC(=O)C(C)c1ccco1 C(=O)(CC(C)(C)C(F)F)NC12C(n3cc(Cn4c(C)ncc4)nn3)CC(CC1)C2 c1(C(=O)NCCCN(C2CCCC2)C(c2cc(C)[nH]n2)=O)cc2c(s1)CCSC2 N1(C(COC(C)(C)C)=O)CCC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C12CCCC2 C1(C)(CC)CCC(C(=O)N(CC(C)(C)C(=O)NCC(C)(C)n2cccn2)C)O1 C1(C)(N)CCC(C)C1.CCC(=O)NCCOC.C12(CC1)C(=O)N2 Cc1csc(C(=O)NC(C(=O)NC2CC3CC3C2)C2CCC2)c1C c1(N(CC=C)CCC2CCC(C)CC2)ccc(S(=O)(=O)N2CCOCC2)cc1F C1(CNC(CCc2scc(C)n2)=O)CCN(C(=O)C(C)c2cc[nH]n2)C1(C)C Cc1ccc(C(=O)N(CC(C)NC(=O)C(C)(C)O)C)c(F)c1Cl Cc1nocc1C(=O)NCC(C1CCOC1)NC(c1cnoc1C)=O c1(C(CNC(c2occc2NCc2nonc2C)=O)NC(C)=O)ccc(Cl)cc1 c1(C(=O)NC2CC(N(C)C(C3CC3(Cl)Cl)=O)C2)cc2c(s1)CCCNC2=O c1(C(=O)NC(C2(O)CCN(C(=O)CC(C)(C)C)CC2)C)cc2cccc(Cl)c2[nH]1 c1(C(=O)OC(C(=O)NCC(c2ccccc2)CC)C)ccccc1.C1CC1 c1(C(N2CC(C(C)NC(C3(C)N(C)CC(OC)C3)=O)C2)=O)n[nH]c2c1COCC2 C1(CNC(=O)NC(C)CN2CCOCC2)Cc2ccccc2C1C C1(C(=O)NC2C(C(N3CCC(SC)CC3)=O)CC2)CC2(CCC2)CO1 Cc1ncc(NC(C2CC2C(C)NC(c2cccnn2)=O)=O)c(C)n1 c1(NCC(N(C(C2CN(CCC)C(=O)C2)=O)C)C2CC2)cnc(C#N)c(C#N)n1 c1(CN(C)CC)cccc(C#N)c1.C1(=O)CCC(=O)N2CCOC(C2)N1 N1(C(C2CC23CCC3)=O)C2CCC1CC(c1cn(-c3ccccc3F)nn1)C2 C1(CN(C)C(C2CCCO2)=O)CCN(C(=O)CCNC(=O)C(F)F)C1 Cc1ncnc(O)c1C(=O)NC1CC(C)(CNC(C23CCCC2CCC3)=O)C1 C1(F)(C(N(C2CCN(C)CC2)C)=O)CCCN(C(=O)C=CC(F)F)C1 C1(NCC2C(C)(C)OCC2)CC2CC1CC21CC1 N1(C(COC(C)=O)=O)CCOC2(CCC(NC(c3cnc(C(C)C)[nH]3)=O)CC2)C1 C1(CN(C(C(OCC)OCC)=O)C)COCCN1C(=O)CCN1CCC1 CC(O)CCCCCC(=O)NCC1CCC1NC(c1ccc2nc(O)[nH]c2c1)=O N1(C(c2scc(C)c2C)=O)CC2CCC1CC2NC(C1CC1c1ccccc1)=O C(=O)(C(CC1CNC1)NC(=O)OC(C)(C)C)NCC#C C1(C(=O)NC2(n3ccnn3)CC2)(OCC)CN(C(C2(C)CC(=O)C2)=O)C1 C(CNC(N)=O)(C(C)C(C)C)NC(C1(SC)CC1)=O.C1(CC)CC2CC1NC2=O c1(CC)cc(C(N2CCCC(NC(=O)C(O)CC(C)C)CC2)=O)cc(F)c1 c1(C2(C)C(C(=O)NC3CC(CNC(C4C(OC)C4)=O)C3)C2)ccccc1F C(=O)(C(Cn1cncn1)NC(c1ccon1)=O)NC1(C(C)(C)O)CCC1 N1(C(c2cc(C)no2)=O)CCC2CN(C(C3CCc4nncn4CC3)=O)CC2C1 c1(C(=O)NCC(CC)NC(=O)CCc2nccs2)cc(N)cc(N)c1 C1(CNC(C(=Cc2cccs2)C)=O)CCCN(C(c2oc(C3CC3)nc2C)=O)C1 C(CCN=C(NCC(=O)OC)NC1CN(Cc2c(C(F)(F)F)cnn2C)C1)OC C(=O)(C1=C(C)CCC1)NC1CN(C(c2c(C)nc(OC)s2)=O)CC1CC1CC1 c1(C(=O)NC2C3C(C)N(C(=O)CNC=O)C2C3)cnc2c(F)c(F)ccc2c1 C1=C(CN=C(NCC2CCOC2)NC2CC(n3ccnn3)C2)CCOC1 CC(CCC(=O)N(C1CCN(C(C2CN(CP(C)(C)=O)C2)=O)C1)C)S(C)(=O)=O c1(N2CC3N(C(=O)Cn4cccn4)C(C3)C2)ncnc2c(F)cccc12 C1(C(=O)NCC2N(C(c3cnc(C)[nH]3)=O)CC=C2)CCC(NC(N)=O)CC1 c1(-c2nnc(N3CC(C)C(C(=O)OC(C)(C)C)CC3)n2C)n[nH]c2ccccc12 Cc1cc(Cl)ccc1CC(=O)NC1CCN(C(=O)CCN(C)CCO)C1C Cc1c(C(=O)NC2CCN(C(=O)C(C)Sc3ncccn3)C2)cccc1[N+](=O)[O-] C(=O)(CCCCCC)N1C(Cn2cc(CCOC(C)C)nn2)CC(CC)C1 N1(Cc2ccc(C)cc2Br)CC2(CN(C(=O)CCN(C)C)CC2C(=O)O)C1 N1(C(CC(CC)C)=O)CCCCC2C1CCCN2C(c1cnc(O)n1CC)=O C1(=O)C(F)CC2CN1C2.C(=O)(C(CN(C)C)N(C)C)N1C(C(=O)NC)CC1 N1(C(=O)CC(C(F)F)n2ccnc2)CC2CCN(C(=O)C3CC3)C2C1 c1(OC)cc(CN2CCC(O)C2C(N2CCOC(O)C2)=O)ccc1Cl C1(CNC(C(C)=C2CC2)=O)CN(C(=O)Cn2ncccc2=O)CCO1 Cc1sc(C(=O)NC(C(C)NC(c2cc(O)ncn2)=O)C(C)C)cc1[N+](=O)[O-] c1(C(=O)NCC(C)(O)CNC(C2CN3CCN2CC3)=O)ccc(C2CC2)cc1 CCCCCCCCC(C)C(=O)N1CCC2(NC(c3cc[nH]n3)=O)CCCC12 C(C(N=[N+]=[N-])C(=O)NCC1CCCCC1C(=O)NCC1(N(C)C)CCC1)OCC C(=O)(C#CC(=O)NC(c1ccc(OC)cc1)CNC(C1(Cl)CC1(C)C)=O)N(C)C C(C(CC(=O)N1CC(C)(NC(c2cccc3scnc23)=O)C1)C(F)(F)F)N(C)C C(C)(CCCCN=c1nc2[nH][nH]cc-2c(O)n1)NC(c1cnc(C)o1)=O CN1CCc2nc(O)c(C(=O)NC34CCCN(C(C5CC(O)C5)=O)C3C4)cc2C1 C1(NC(c2c(OC)csc2)=O)CC(C)N(C(c2cnn(CCF)c2)=O)C1 CCC(C)(CNC(=O)Cc1cnn(C)c1)C(=O)NCC(C)(C)CN(C)C c1(CCCC(N2CCC(O)(CNC(CS(CC)=O)=O)C2)=O)nc2ccccc2s1 C1(CNC(CC2CCN(C)CC2)=O)CCCN(C(=O)CC2COCCO2)CC1 C1(NC(c2cc(C)c(C)s2)=O)CCCCCN(C(c2ccc(CCF)cc2)=O)C1 c1(C(N(C2CCC(NC(CCCC#C)=O)CC2)C)=O)cc(C)c(N)c(C)c1 c1(C(=O)NC(CNC(C(C)OCC(F)(F)F)=O)C2CCC2)cnn2ccncc12 C(CCCCC(=O)N(C)CC1COCCN1C(=O)CCc1cnoc1)=CC N1(C(c2cc(Br)cc(Cl)n2)=O)CC(CO)C2(CCC2)C1 Cc1ccc(F)c(CC(=O)NC2CC3CN(C(c4nc(C)no4)=O)CC23)c1 CC1CCCC=C1c1cscc1NC(c1cc(F)ccc1I)=O N1(C(CC(CNC(C(C)(C)CCF)=O)O)=O)CCC12CCCSC2 C1(CC)CCN(C(c2ccn(C)n2)=O)C1C(=O)NCCN(CC)CC Cc1cc(C(=O)NC(CCF)C(=O)NC2CCCOC2)cnn1 c1(CCC(=O)NCCN(C(CCN(CCC)C)=O)C)ccc(F)c2ccccc12 c1(C(C(=O)NC(CC(C)NC(=O)CC23CC(C2)C3)C)(F)F)ccc(F)cc1 c1(C(=O)NC2CCCN(C(C(C)=C3CCCC3)=O)C2)cc(C)nc(C)c1O O=S(=O)(c1cccnc1N1CCC(CC(F)F)CC1)NCC1CCC2(CC2)CO1 C1(NC(c2cc(C(C)C)[nH]n2)=O)CCCCC1NC(C12CC(C)C1C2)=O c1(OC)ccc(C(N2CC(NC(c3cc(C)co3)=O)CC2C)=O)c(OC(C)C)c1 c1(C(=O)NCC(C)(C)CNC(=O)C=CC2COC(C)(C)O2)ccn2nccc2n1 N1(C(C(CC#C)C)=O)CCCN(C(=O)C(c2c(F)cccc2F)(C)C)CC1CO C(=O)(CC(CNC(=O)CC1(C#N)CC1)C1CCC1)N(CCN(C)C)CCO C1(C)(C(N(C)CCn2cccn2)=O)CN(C(=O)CC2COCC2O)C1 c1(C(=O)NCC=CCC(N2CCC(C(C)(C)O)CC2)=O)c[nH]c2nccc-2c1 c1(CCC(=O)NC2C(C)CN(C(C3(O)CCOC3)=O)C2)nc2cccnc2[nH]1 CC(C(=O)NCC1(F)CC(NC(c2ccnc(S)c2)=O)C1)C(C)(F)F N1(C(c2c(C)oc(Cl)n2)=O)CCN(C(c2cc(O)ncc2F)=O)CC(O)C1 Cc1cccc2c1CC(C(=O)NC1COC3(C1)CN(C(C14CSC(C1)C4)=O)C3)O2 c1(C(C)C)ccc(F)c(C(=O)NCC2CN(C(C3(OC(C)=O)CC3)=O)CC23CC3)c1 c1(OC)cc(Cl)c(Cl)cc1C(=O)NCc1ncsn1 c1(C(=O)NC(CCCNC(CCCC#C)=O)C)cc(O)ccc1F c1(C(=O)NC(CC)(CNC(=O)C(C)OCC(C)C)CC)cc(Cl)cc(Cl)c1N c1(C(=O)NCC(CNC(=O)C=CC=C(Cl)Cl)OC)nc2ccc(C)cn2c1N N1(C(c2cn(C(C)C)nc2)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC1CO Cc1cc(C(=O)NC(c2ccccc2)C(N2CC(O)(c3nn[nH]n3)C2)=O)nc(O)c1 c1(C(=O)NCCC(CNC(C2(CSC)CCC2)=O)O)cc(F)c(F)cc1F C1(C(=O)NC(CCN(C(C(C)c2ccsc2)=O)C)C)(C2CC2)CCCO1 C1(C(=O)NCC(CC)NC(c2cc(C(C)C)on2)=O)CCCN1C(C)=O c12ccc(Cl)cc1SCC1CCN(C1)C2=O.CCC(C)OCC(=O)N(C)C(C)C CC(C)CC(C)(C)C(=O)N(CC(O)CN(C(=O)C(C)CCc1ccccc1)C)C C1(NC(c2ncoc2C(=O)NCCO)=O)CCCN(C(C2CC23CCC3)=O)C1 Cc1ccc2cc(C(N3CCCCC3C(=O)NCC(=O)C3CC3)=O)c(F)nc2c1 c1(CC)cc(C)ccc1C(=O)N(C1CC(NC(C2SCCC2C)=O)C1)C C1(C(C)(C)C)CN(C(c2ccc(O)nc2Cl)=O)CCN1C(C1CCNC1=O)=O C12(C(NOC(C)C)=O)CCC(CC1NC(C1CCCC3(CC3)C1)=O)C2 c1(NC(=O)C=CCF)ncnc2sc3c(c12)CCC3.CC1CC2CN1C2 c1(C(C)NC(C(CC)n2cc(CCOC)nn2)=O)ccc(C)c(Cl)c1 CCC(CC(=O)NCC1CC(F)(CNC(C2C(C)(C)C2(C)C)=O)C1)C(C)(C)C c1(C(=O)NC2C(NC(Cc3cc(C)on3)=O)COC2)cn2ccc(F)cc2n1 Cc1cc(C(=O)N(C2CN(C(c3cnn(CC(F)F)c3)=O)C2)C)cc(C)c1F C(=O)(CCCCC(C)=O)NC1C(NC(c2ccc(OC)cn2)=O)CCCC1 Cc1cccnc1C(=O)NC(C)C(C(C)C)NC(c1ncccc1N)=O C12(C(=O)NC(CNC(c3n(CC)nc(C)c3)=O)CO)CC3CC(C1)CC(C)(C3)C2 C(=O)(C1CCCc2c[nH]nc21)NCCC(CCNC(c1nc(C)sc1)=O)C N1(C(C=Cc2c(C)csc2)=O)CC2CCN(C(C3CC34CC(O)C4)=O)CC2C1 C1(NC(C2(CC)CCCO2)=O)CCCC(CNC(c2cccnc2C)=O)C1 n1(CCN(C(C)C(F)(F)F)CC(=O)OCCSC)ccc2cc(Br)ccc12 C1(CNC(C2C(CC)OCC2)=O)CC2(CC2)CN1C(c1ccc(C#N)[nH]1)=O c1(C(=O)NC2(CC(N3CC4C(C(C)(C)O)C4C3)=O)CC2)ccn2nccc2c1 CC#CCCCC(=O)NCC#CC(=O)NCC1(CSC)CCCC1 CN1CCC(O)(CC(=O)N(CCN(C(=O)C(F)C(C)(C)O)C)CCO)CC1 Cc1cc(N)c(C(=O)N(C2CCCC2)CCCNC(c2ccncc2)=O)nc1C c1(C(N2CC(O)(C(C)NC(=O)CCc3ncco3)C2)=O)ccc2ccn(C)c2c1 N#Cc1ccsc1C(N1CSCC1C(N1CCC(n2cncn2)C1)=O)=O c1(CNC(CC2(CNC(C(C)(C)OCCC)=O)CC2)=O)c(C)cccc1Br C1(NC(COCC)=O)CN(C(c2cc(=O)c(OC)c[nH]2)=O)CC2(CCC2)C1 N1(C(C2CCC(CC)O2)=O)CCC2(C1)CN(C(c1cccc(N=[N+]=[N-])c1)=O)C2 Cc1nn(C)cc1CC(=O)NCCc1n[nH]cc1C(=O)NCC1CC(O)C1 c1(C(N(C2CCCCC2C(N)=O)C)=O)ccccc1Cn1cc(Br)cn1 CN(C)NC(=O)CCC(=O)NCC(O)CC(=O)N1CCC(O)(CO)C1 C(CCNC(C1CCCSC1C)=O)(C(C)C)NC(C=CC)=O C=C(C)CCC(c1nnnn1Cc1ccccc1)NCCc1cccnc1OC n1(CC(=O)NCC(C)(CC(C)C)NC(C(CCSC)O)=O)c(C)cc(C)nc1=O c1(CO)ccnn1C.C1(C(=O)NCCOCCNC(=O)NC2CC2)(CC)CC1 c1(SC)ccsc1C(=O)N(C)CC1CCCN1C(=O)CC1CCCC1C CC1CCCC(OCC(=O)NC(CNC(c2cc(CCO)on2)=O)C2CC2)C1 C1(NC(C(N)=O)=O)COC2(C1)CN(C(C1(C(F)(F)F)CC=CCO1)=O)C2 c1(CC(=O)N(CC(C)NC(=O)C(C)CF)C)cc2ccccc2o1 N1(C(CCC(C)NC(c2c(C)csc2)=O)=O)CC2CCC(C1)N2C CC1CC(NC(C2CCCC23CC3)=O)CCN1C(c1cnn2ccsc12)=O C=CCCC(F)(F)C(=O)N1CC2CC(NC(C3CCCC3F)=O)C(C2)C1 N1(C(C2(C(C)(C)F)CCC2)=O)CC2CC1C2NC(=O)CN1CCCCC1 C1(CNC(CN(c2cnccn2)C)=O)CN(C(=O)CC2CCC2)CCN1C c1(OC)c(CN2CCCC(C)(C(N3CCC(NS(C)(=O)=O)C3)=O)C2)c(C)nn1C c1(C(N2C(C(N(C(CC)COC)C)=O)CC=CC2)=O)cnc(O)cc1C c1(C(=O)NC2C(NC(C34CC(C)(C3)C4)=O)C2)cc(Br)cc(Cl)c1F N1(C(=O)NCC(c2ccccc2)CC)CC2CN(C)CC2C1 N1(C(C(C)S(C)(=O)=O)=O)CCC(NC(=O)C2=CCOC2)C(CO)CC1 N1(C(=O)NCc2n(CC)nnn2)CC2CC(N3CCC(OC)C3)C1C2.C(=O)O c1(NC)scnc1C(=O)N(C(C)CNC(=O)CC1CCC(=O)N1)C C1(C(=O)NCCNC(c2ccc(O)nn2)=O)CCC(O)CN1NC(N)=O N1(C(C2(c3cccc(C)c3)CC2)=O)CCN(C(=O)CC2CC=CCC2)CC(C)C1 N1(C(COCC=C)=O)CC(NC(=O)C=Cc2nonc2C)CC(O)C1 C(=O)(CCS(=O)(=O)c1ccccc1)NC(C)CC(C)NC(=O)CCC(N)=O c1(C(=O)NC(C(C)C)(C)CNC(C2CCCOCC2)=O)ccc2c(c1)OCC2 N1(C(C2(C)CCC(C)C2)=O)CCC(C(=O)NCC2CCC=CO2)C(C)C1 c1(C(N2CCC(C)C(N(C(=O)Cc3ccco3)C)C2)=O)cc2cccnc2cn1 N1(C(Cc2c(C)noc2C)=O)CCOC2CN(C(C3CCCC(F)(F)C3)=O)CC12 c1(CC)ccc(C(=O)NCC2(NC(c3cncc(F)c3)=O)CCOC2)cc1CC C1(C)(C(N(CCCCCNC(c2cc(CC)sn2)=O)C)=O)CC(OC)CN1C c1(C(N2CCCC(n3cc(C4(O)CCOC4)nn3)C2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(C(CC2CCCC2)NC(CCSC)=O)=O)CC2(CO)CCC1CC2 N1(CC)CC(C(=O)NC2(C)CC(NC(=O)Cc3ccc(F)cn3)C2)CC1=O N1(CCC)CC(C(=O)NCC=CCNC(=O)CC2CCCC2)CC1=O CN1CCC(NC(=O)C(=O)Nc2cc(Br)cnc2S)CC1=O c1(OCC)cnc(=NCC2CCC(NC(c3ccc(C)c(OC)c3)=O)C2)[nH]c1 C1(CNC(=O)COc2ccon2)(CO)CCN(C(=O)CCCCC2CC2)CC1 c1(COCC(=O)NCC(C)CNC(=O)CNC(N)=O)cccnc1 C(CO)(CCCCNC(c1cc(C2CC2)cs1)=O)NC(c1c(SC)cn(C)n1)=O C1(NC(CC2CC(OCC)C2)=O)COCC1CNC(c1ccoc1C)=O N1(C(=O)OC)CCC(C)C(CNC(C2(n3cc(CN)nn3)CCC2)=O)C1 c1(C(=O)NCC(CN(C(=O)C(C)(C)C(F)(F)F)C)(C)C)cn(C)c(=O)nc1O C1(NC(C(C)C(C)O)=O)COCCN(C(=O)CCCC(O)c2ccccc2)C1 C1(NC(=O)COC)CCCC1CNC(C1CCCC1)=O.c12ccc(s1)[nH]c2=O.CO C(C(N=c1[nH]c(C(C)(C)C)nc(=N)[nH]1)C(C)C(C)C)NC(C(CC)CC(C)C)=O Cc1cc(C(=O)N(C)CCOCCNC(=O)Cc2nccs2)[nH]c1C c1(CC)cncc(C(N2CCC(NC(C34CC(C)(CO3)C4)=O)CC2)=O)c1 N#CC1(C(=O)NCC(O)CNC(=O)CSCCc2ccccc2)CC=CC1 CCCCC(O)CC(=O)NCC(C)C(F)C(=O)NCc1cnc(C)s1 N1(C(C(=O)NCC(F)F)=O)CCC2CN(C(=O)C(F)(F)C(O)C3CC3)CCC12 c1(C(=O)NC2CC(NC(C(CC(C)(C)C)O)=O)C2)cc(O)c2ccoc2c1 N1(C(=O)CC2CCSC2)CCC2(CC2C(N2CCC(O)C2)=O)C1 CCC(CC)C(C(=O)N1CC(C)CCC1C(N1CC(S(C)(=N)=O)C1)=O)OC N1(C(CC2CC(=C)C2)=O)CC(NC(c2cnc(C3CC3)o2)=O)C2CC12 c1(CC(=O)N(CCCOCCNC(C2CC(COC)C2)=O)C)ccc(C)c(C)c1 N1(C(C(C2CN(C(=O)C3=CCC(C)CC3)C2)OC)=O)CCN2C(=O)CCC2C1 N1(C(C(C(C)C)NS(N)(=O)=O)=O)CCC(C)N(C(c2cn(C(C)C)nn2)=O)CC1 N1(C(C2N(C(C(CCCC)F)=O)CCC2)=O)CCOCC(C2CC2)C1 C#CC1(O)CC(C(=O)NCC2(C)CCN(C(c3ccnc(OCC)c3)=O)C2)C1 c1(C(N2CCC(CNC(CC3(O)CCCN(C)C3)=O)C2)=O)cnc2c(c1)CCC2 C(=O)(C(F)C(F)(F)F)NCCCN(C(C1N(C(CC)=O)CCCC1)=O)C c1(CO)ccc(F)cc1Cl.N12CCN(CC1Cc1cccnc1Cl)NC(=O)C2 c1(-n2cc(CCNC(C3CC(O)C(F)C3)=O)nn2)cccc(Cl)c1 c1(N2C3CN(C(Cn4c(=O)ccc(C)c4)=O)CC2CC3)nc(C)cc(C)c1C#N C(=O)(CCCCC(=O)NCC1CN(C(c2n[nH]c3c2CC2CC32)=O)CCO1)NC C1(C(=O)NC(CC#C)CO)CCC2CCC1N2C(=O)Cc1ccccc1O C1(CCNC(c2cc(C)c(C)[nH]2)=O)CCN(C(c2cc(=O)cc[nH]2)=O)C(C)C1 c1(C(N2CC(C(=O)NC3(CC(=O)OCC)CCCC3)C2)=O)cccc(CO)c1 C1(NC(CSc2nc(C)cc(C)n2)=O)CC2(NC(=O)Cn3cccc3)COC1C2 C1(NC(=O)C=CC2CCC2)CN(C(=O)CC2CC2)C2(CCOCC2)C1 C=CCC(CC)C(=O)NCCCN(C(=O)C(c1ccc(OC)cc1C)C)CCC c1(C(=O)NC(CC(C)C)CNC(C2CCC(C)(C)C2)=O)cc([N+](=O)[O-])nn1C c1(C(N2CCC(COC)(NC(c3conc3C)=O)C2)=O)cc2cccn2c(O)n1 N1(C(c2c(CC)ncs2)=O)CCCN(C(=O)Cn2nc(C)oc2=O)CC1 C1(C(N2CC(C(N)=O)(CNC(=O)C(F)OC(F)(F)F)C2)=O)CCC2(C1)CC2(F)F c1(C(=O)NCC(C)N(C(=O)CCNCC(F)F)CC)c(N)sc2c1CCC2 c1(C(=O)NC2CC(CNC(C3(COC)CCC3)=O)C2)ccnc(F)c1OC c1(C(=O)NC(C2CCN(C(=O)Cn3cnnc3)C2)C)cnn2ncccc12 N1(C(c2cncs2)=O)CCCC2(CCN(C(C3CCC3(F)F)=O)C2)C1 N#Cc1cn(CCC(=O)NCC2CCCN2C(C2CCOCC2)=O)c(=O)nc1O CC(C)(C)C#CC(=O)N1CCCCC(CNC(=O)CCC2CCCC(=O)N2)C1 N1(C(C2CCC(NC(=O)OC)CC2)=O)CC=C(CCNC(C2SCCS2)=O)CC1 C#Cc1cc(C(=O)NC23CC(NC(c4cnc(SC)nc4Cl)=O)(C2)C3)ccc1C C(C(C)(C)C(=O)OC)N(C(C1CC12CN(C(=O)Cc1ccn(C)n1)C2)=O)CC Cc1cn2ccnc(C(N3CC=C(CNC(C4COC(C)C4)=O)CC3)=O)c2n1 N1(C(CC=C)=O)CCCC(NC(c2n[nH]c(O)n2)=O)C1C C(=O)(CCCCN=[N+]=[N-])N1CC(N2CCN(C(C(C(C)C)OC)=O)CC2)C(C)C1 CCC(C)CCCCC(=O)N(C1(CCCC(N2CCC(C)C2(C)C)=O)CCC1)CC N1(C(=O)OC(C)(C)C)CCCC1(C)CCCNc1cnn(CC2CCCOC2)c1 C(C)(N=c1nc(N2CCc3n[nH]cc3C2)c2c([nH]1)CSC2)c1nc(C)sc1 N1(C(c2cn(C)nc2Cl)=O)CC2CN(C(C3CC(C)(C)CO3)=O)CC2(C)C1 N1(C(c2nc(SC)sc2)=O)CCN(C(C2CCS2(=O)=O)=O)C2(CCC2)C1 c1(C(N2CCC(N(C)C(c3cc(C#N)cs3)=O)C(F)C2)=O)cc2cccnn2n1 N1(C(Cc2c(C)con2)=O)CC(NC(=O)C(F)(F)c2csc(=N)[nH]2)C(C)C1 C1(C(C)NC(=O)COc2ccn(C)n2)CCN(C(=O)C(F)CC2CCOC2)CCO1 C1(=CC(=O)NC(CSC)C)CCN(C(=O)C=C(C)C2CC2)CC1 CCC(O)C(C)C(=O)N1CCCC(CN(C(=O)CCS(C)=O)C)C1 N1(C(C2CCN2Cc2ccc(O)c(Br)c2)=O)CCc2ccc(Cl)cc2C1 C#CCCC(O)CCNC(=O)CCCCN(C(=O)COC1CCOC1)C c1(C(N(C)CC2CCCN(C(c3ccc(C)o3)=O)C2)=O)noc2c1COCC2 N1(C(CCC)=O)CC2(CC(NC(=O)CC3CSC3)C2)C1 c1(C(N2CC(CNC(C3(C4CC4)CCC3)=O)CC(C)C2)=O)cn(C)c(=O)nc1O C(C)(CO)(C(=O)N(C1CC2(CCC2)C1)C)NC(C(CC)NC(C)=O)=O Cc1cc(C(=O)NC2CN(C(=O)C(Cl)(Cl)Cl)CC2O)cc(O)c1 C1(C(=O)NCCCOCCN(C)C(C2(C)C=CCC2)=O)CCc2ccccc2O1 O=C(C1=CCOC1)NC1(c2ccccc2)CCN(C(c2ccc(NC)cc2)=O)C1 C1(NC(C2(CNC(=O)CC3CCC3)CCCO2)=O)CCc2nncn2C1 C1(C(=O)NC(CCNC(c2cnns2)=O)Cc2ccccc2)COC2COCC12 N1(C(c2nc(NC(C)=O)sc2)=O)CC(NC(c2snc(Cl)c2Cl)=O)C(C)(C)C1 C12(NC(Cn3c(C)c(Cl)cn3)=O)CCN(C(=O)C=C(Cl)Cl)CC1C2 C(=O)(C(CC)C(F)(F)F)N1CC(OC2CCN(C(CCC(=C)Cl)=O)CC2)C1 CC1CN(C(C2COCCN(CC(F)(F)F)C2)=O)CCN1C1CCCCC1 c1(CC(=O)N(CCN(C(c2cnnc(O)c2)=O)CC)CC)ccc(F)c(F)c1 C1(NC(C=CCC23CN(C2)C3=O)=O)CC2CCCC2C1.C1(C(N)=O)(CC)CCC1 CC(C)CC(C)CC(=O)N1CCCC(C(N2CC(C)(CCO)C2)=O)C1 C(=O)(C(C)C(C)NC(=O)C1CC1)N(CC(=O)NC)C C1(C(N(CCC)C(C)C)=O)C2CC(O)C(C2)N1C(C1CC1(C)C(F)F)=O C1(CCNC(CC(C=C)C)=O)CN(C(c2nn[nH]c2Cl)=O)CCCO1 C1(COC)CN(C(=O)CCSC)CCN1C(=O)CCC1CCCO1 C(=O)(C(CC#CC)NC(C1CC(CC)C1)=O)NC(CC#C)C c1(C(=O)NC(C(=O)NCC2CC2)C2CCCC2)cccnc1 c1(CC(N2C(C(=O)Nc3cccc(N(C)C)c3)CC(=C)C2)=O)c(F)cccc1Br Cc1c(C(=O)NC(C)CNC(c2ccc[nH]2)=O)sc2ncnc(N)c12 c1(CC)ncoc1C(=O)NC(C)CC(C)NC(=O)C(C)CC1CCCCC1 c1(C(=O)NC2C(NC(C(C(C)C)F)=O)CCC2)ccc2c(c1)COCC2 c1(C(=O)NCC2CC(NC(c3c(OC)oc(C)n3)=O)C2)cc(C#N)ccc1N c1(CC(N2CCC(CC)C2)=O)cc(-n2cc(C(C)(C)O)nn2)c(C)o1 c1(C(=O)NCCN(C(c2c(C)onc2CO)=O)C2CC2)cnc2c(c1)nnn2C c1(C(N2CC(CNC(C(C)(C)OC)=O)C(F)(F)C2)=O)c[nH]c2cc(F)c(F)cc12 N1(C(C(c2ccc(C)s2)C)=O)CC2CC(NC(=O)C=Cc3ccncn3)CC2C1 C1(CC=C)CCCC1(c1nnnn1C(C)C)NCCCn1ncnc1CNC C1(CNC(Cc2ncc(C)s2)=O)CCC(NC(C23CC(C2)C(C)O3)=O)CC1 O=C(C(F)C1=CCCCC1)N(c1ccc(Br)cc1)S(=O)(=O)Cc1ccon1 C1(NC(=O)CC2CC2(Cl)Cl)CN(C(=O)COc2cccc(O)c2)CCC1(F)F c1(-c2cnc(NCc3c(C)cc([N+](=O)[O-])cc3)c(C)c2)ccc2c(C)c[nH]c2c1 N1(C(c2c(C)cc(C)s2)=O)CC(C(=O)NCCC(C)N2CCCC2)C2(CC2)C1 Cc1ccc(C)c(OCCNC(C2(C)CC(O)CN2C(=O)C(C)NC=O)=O)c1 C(c1c(F)ccc(Cl)c1F)=CC(=O)NCC(F)CNC(c1cc[nH]n1)=O CC1Cn2nccc2CN1C(=O)CCCCN(C(=O)CCC1CCC(=O)C1)C CS(=O)CCC(=O)NCC(CO)NC(=O)CNC(=O)CCCCO C1(NC(C(CSC)O)=O)CC2(C1)CN(C(=O)CCc1ccc(C)s1)C2 N1(C(C2C3(CC(NC(COCCCCC)=O)C3)C2)=O)CC(S(N)(=O)=O)C1 N1(C(C(C=CC)O)=O)CCN(c2nc(COCC)ns2)CC(O)C1 c1(C(=O)NC(C2N(C(CS(CC)=O)=O)CCC2)C)cc(C2CC2)n(C)c1C C1(NC(C(CC)=CC)=O)CC2CC(NC(C3CC34CC(OCC)C4)=O)C2C1 C1(NC(c2nc(CCC)oc2)=O)C2CC3CN(C(=O)CS(=O)(=O)NCC)C1C3C2 Cc1ccc2nonc2c1C(N1CC(CNC(C2CN(C(N)=O)C2)=O)C(C)C1)=O c1(C(N2CC3C(CNC(C4(CC#C)CC4)=O)(C3)C2)=O)cc(C)ccc1Cl C1(CNC(=O)Cc2cnoc2)COCCN(C(c2nocc2Br)=O)C1 CC1CCN(C(=NCCF)NCC2C(F)(F)C23CCC3)CC1 N1(C(c2c(OC)noc2C)=O)C(C(=O)NCC2CCC(C)(C)O2)CC2CCCC12 C1(CC=C)(NC=O)CCCC1.c1(C(=O)OCCCNC(=O)CCC)cc(CC)c[nH]1 c1(C(=O)NCC2(CCNC(c3c[nH]nc3Cl)=O)CC2)cc(NC)ccn1 c1(NC(c2cc(C(CC)C)no2)=O)ccc2c(c1)NC(=O)CCC2 c1(CC)cncc(C(=O)OCC2CCCN2Cc2ccccc2)c1 c1(C(=O)NCCS(=O)(=O)N2CCOCC2)cc2ncnc(O)c2cc1Cl c1(NC(C2CCC(Cc3ccccc3)C2)=O)nccnc1C(F)(F)F c1(C(=O)NCC(CC)NC(=O)CC(O)CN(C)C)cc(CO)oc1C C1(COC)CN(C)CCN1C(=O)CCC(C)n1cc(COC(C)=O)nn1 c1(C(=O)NCC2N(C(c3nc(C(=O)OC)oc3)=O)CCC2)ccc2c(c1)CC2 N1(C(C2(C)CC(F)C2)=O)CCCCC1CCNC(=O)Cc1ccnc(O)c1 c1(CNC(C2(C#C)CC2)=O)cc(C(=O)NCC2CCOC(C)C2)ccn1 C(CC)(CCCCC)(c1n(CC(=C)C)nnn1)NC1(CS(C)(=O)=O)CC1 c1(NC(C2CC(NC(c3cc(F)ccc3O)=O)C2)=O)ccc2c(n1)CCC2 Fc1cc(CNCC2CCCC2c2ccccc2Br)ccc1Br C(=O)(CC(F)(F)C(F)F)NCC1C(NC(C=CC=CCC)=O)CCC1 c1(C(=O)NC(CN(C(=O)CCC(C)C)CC)C)cnc(-c2ccncn2)nc1O Cc1ccc(C(C)NC(=O)C(C2CCN(C(C3(C(=O)C4CC4)CC3)=O)C2)F)cc1 N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CC(NC(c3cn4ccsc4n3)=O)CC1C2 c1(OCC)cc(Br)ccc1C(N1CCOC(CNC(c2cncs2)=O)C1)=O CC1C(O)CCCN1C(C1CCCN(C(=O)CCCC2CCCO2)C1)=O C1(COC)(CNC(C2CC(C)(NC(=O)C(F)C3CCC3)C2)=O)CCCC1 c1(CC(=O)NCCC)c(C(=O)N(CC(=O)N(C2(C(C)C)CC2)CC)C)n[nH]c1CC C(C(C)(O)C(F)(F)F)N(C)C(=O)NCC1(F)CCOC1 C1(N(CC(C(F)F)n2cccn2)CC(F)F)CCCC2(CC1)OCCO2 C1(C(N2CCCCC(C(CC)CC)C2)=O)CC2(CCN(C(=O)C[SH]=CCO)C2)C1 c1(CC)ccc(C(N2CC(C)C2C(=O)NCC2CC2(F)F)=O)cc1 C=C(Cl)CCC(=O)NCCOC1CCN(C(c2nc(-c3ccco3)oc2C)=O)C1 c1(OC(C2C(NC(C=CCC)=O)C2)=O)cc(C)ccc1C(=O)NCC1CC1 N1(C(C(CCCOC)NC(c2cscc2C)=O)=O)CC(C)CC(F)(F)C1 CS(=O)(=O)c1cc(-c2nc(-c3ccc4cncn4c3)nn2CCF)co1 Cc1cc(Cl)ccc1C(=O)NCC1CC2CCC1N2C(=O)CC1CC1(Cl)Cl c1(C(N2CC(O)(CNC(c3cccc(O)c3)=O)C2)=O)ccc(F)c2occc12 C1(CCCNC(CC(C)OC)=O)CCCCN1C(c1cccnc1C)=O N1(C(c2c(C)[nH]c(=N)s2)=O)CCCN(C(=O)C(N2CCOCC2=O)C)C(C)C1 C(C(=O)N1CCC(C)(NC(=O)CCc2cccs2)C1)(C(C)C)SC CC(C)(C(=O)O)C(CCO)N1CCC(C(=O)NCCc2n[nH]c(=N)s2)CC1 C1(CNC(C2CCC(CC)O2)=O)CCN(C(=O)CC2(C)CCCCC2)C12CC2 c1(C(=O)NCC2(F)CC(NC(C3CCC(C)C3)=O)C2)ccc(S(N)(=O)=O)cc1F CCC(CC(=O)N1CCCC(O)(CNC(c2ccc(C(F)F)o2)=O)CC1)C(F)F N1(C(C2N(C(c3ccc(OC(C)=O)cc3)=O)C(C)CC2)=O)CCCC(C#N)C1 c1(C(=O)NCC2CN(C(CCCn3c(C)ncc3)=O)C2)cc2oc(C)c(C)c2[nH]1 C1(NC(c2cc(CCC)on2)=O)CCC2CC1CN2C(c1cnccc1CC)=O C(=O)(C(C)CCC(C)(C)C)N(CCN(C(C)C)C(C12CC(CO)(C1)OC2C)=O)C c1(C(=O)NCC(CN(C(Cc2c(C)ocn2)=O)C)C)cc2c(nc1O)CCCC2 C1(NC(c2nn(C)c(C3CCCO3)c2)=O)COC2(C1)CN(C(c1cocn1)=O)C2 c1(C(=O)NCC(N(C)C)C2CC2)cncc(CNC(=O)CCCN(C)C(C)C)c1 c1(C(=O)NC(CC)CNC(C2CCCOC2C(C)C)=O)ccc2c(n1)NCC2 c1(C(N2CC(CNC(C(C)C)=O)C(C(F)(F)F)CC2)=O)nc2c(s1)COCC2 Cc1c(F)ccc(C(N2CC3COCC3(C(=O)NCC3(CN(C)C)CC3)C2)=O)c1O N1(C(c2nc(C)oc2)=O)CCCCC(C2CN(C(=O)CCCCF)C2)C1 N1(C(CCOC)=O)CCC(NC(=O)C(O)C2CN(C(=O)C=CC3CCC3)C2)CC1 CCCCC(O)CC(=O)N1CCN(C(c2n[nH]c(C)c2C)=O)C(C(C)(C)C)C1 c1(OC)cc(I)c(C(=O)OC(C)(C)C)cc1OC.C12CON(C(=O)O1)C2.CO N1(C(CCC=C(C)C)C(=O)NCc2ccccc2Br)Cc2ccccc2C1 N1(C(c2cn(C)nn2)=O)CCC(NC(c2ccnc(O)c2)=O)C(CO)C1 C(N=c1nc2c(ncn2C)c(NC2CCC3(CC3)C2)[nH]1)c1cccc(S(C)=O)c1 N1(CCC(=O)NC2CC(C)N(C(=O)CN(C)C(N)=O)C2)Cc2ccccc2C1=O C12(CNC(c3c(C)cc[nH]3)=O)CC(C1)C(NC(=O)Cc1cn3ccsc3n1)CO2 c1(C(=O)OCCC(c2ccc(OC)cc2)(C)C)ccc(S(=O)(=O)NOC)cc1 C1(NC(CC2OCCN(C(CN(C)C(N)=O)=O)C2)=O)CCn2ncnc2C1 O(C=CC(=O)N1CCCC1CCCNC(c1n[nH]cc1-c1ccncc1)=O)CC c1(C(=O)NCC(CC)NC(=O)C(CC)CC(F)F)c(F)cc(Cl)cc1Cl N1(C(C(CC)c2ccccc2)=O)CCCC(CNC(c2cc(F)n[nH]2)=O)CC1 C1(CNC(C(CC)OC)=O)CCC(N(C(=O)CNC(C2CCCCC2)=O)C)CC1 C(N=c1nc[nH]c2c(F)cccc12)C1C(C)CN(C(c2cc(O)no2)=O)C1 C1(C(=O)NC(CC(C)NC(=O)COCCO)C)CCCCC12CCC2 CC1CCc2c(sc(NC(=O)CC3CCCC4(CCC4)O3)c2C#N)C1 N1(C(c2ccc(OC)s2)=O)CC(C)CC1C(=O)NCCCCC(N)=O c1(C(N(C2CCCC2)CC#C)=O)cnn(CCNC(c2cnc(O)o2)=O)c1 C(CCCCNC(c1ccc(C2CC2)[nH]1)=O)N(C(=O)CNS(=O)(=O)C1CC1)C CCC(CC(=O)N1CC(CNC(=O)CCC(N)=O)C(F)(F)C1)CC(F)(F)F c1(C(=O)NCCN(C(c2cc(C(F)(F)F)ccn2)=O)CC)cc(S(N)(=O)=O)c[nH]1 C(=O)(C(C)(O)CC(F)(F)F)NCC(CNC(CCOCC(C)C)=O)O C1(C(=O)NCCCCNC(C(C)(C)c2cnco2)=O)CCc2cncn2C1 C(=O)(C1=CC2(CN(C(=O)C3=CC4(CCOC4)C3)C2)OC1)NCCCC Nc1c(F)cc(C(=O)NC2CC(NC(=O)Cn3cc(C4CC4)cn3)C2)cc1F n1(CC(=O)NC2CN(C(C3(CCOCC)CCC3)=O)C2)ccc(C)cc1=O c1(NC(C2C(NC(c3cocn3)=O)C2)=O)cc(Cl)ncc1[N+](=O)[O-] Cc1ccc(F)cc1N(C(=O)C(=O)NC(c1ccco1)CO)C C1(O)(CCNC(C2(CC(C)C)CC2)=O)CCN(C(=O)CC2CCC(C)CO2)CC1 C=CC1(NC(N(C(C2C3COCC23)C(=O)NCCSC)CC)=O)CCC1 c1(C(=O)NCC2N(C(c3nc(C(C)OC)sc3)=O)CC2)c[nH]c(C)c(Cl)c1=O c1(NC(CC(=O)Nc2ccon2)=O)ccc(F)cc1.C1(=O)C=CC(OC)O1 C#Cc1cccc(C(=O)NC2CC(CCNC(C3CCC(C)C3)=O)C2)c1F C1(C(=O)NCC(CC)NC(=O)CS(=O)(=O)CC)CCc2ncnc(C)c2C1 CC(C)(C)CC(O)C(=O)N1CCC(C(=O)NC2C=CC(CO)C2)(CO)CC1 C1(C(=O)NCC23C4C5C6C4C2C6C35)CC2CCC(C1)O2 N1(CC2(C=C)CCC2)CC2(CN(C(c3ccn4ncnc4n3)=O)CC(C)(C)O2)C1 C1(CC)(NC(c2ns[nH]c2=O)=O)CCCN(C(=O)C(N2CCNC2=O)C)C1 N1(C(c2cc(C)c(O)nc2)=O)CCC=C(C(=O)N(C2(C)CC2)C)C1 C1(NC(c2c(F)ccc(C#C)c2)=O)CN(C(=O)CCSCC)CC1S(C)(=O)=O C1(CN(C(c2scc(COC)c2)=O)C2CC2)CCN(C(=O)C2=CCOC2)CC1 N1(C(C(=O)NCC2CN(C(=O)CC(C)(F)F)C2)=O)CCN(CCOC)CC1 N1(C(C2CN(C(C)C)C(=O)C2)=O)CCC(C)(C)C1CNC(c1cncc(F)c1)=O N1(C(C(CC)N(C)C(c2cccs2)=O)=O)CCC(OCCNC(=O)CSC)CC1 c1(CC=CC)cccc(C2CCN(C(C3CC(O)(c4ccccn4)C3)=O)CC2)c1 c1(C(=O)NCC(C=C)O)cc(OC)c(OC(C)C)cc1C C(=O)(CC(C)(O)CCC)NC(c1cn(-c2ccc(OCC)cc2)nn1)C c12cc(F)c(cc1F)C(=O)OC2.C1(OC)CCN(S(=O)(=O)C(C)C)CC1 CCCCC(C)CCC(=O)N1CCC(N(C(=O)C(C2CCCCC2)O)CC)CC1 C#CCCCCCCC(=O)N1CCC(C(C)NC(=O)C(C)OCCC=C)CC1 c1(C2C(C(=O)NC(CNC(=O)C3=CCSC3)CO)C2)cccc(F)c1Br C1(CNC(CCN(C(C)=O)C)=O)C2CN(C(c3conc3C(C)(C)C)=O)CC12 N1(C(C2CCCN(C(c3c(CC)ncs3)=O)C2)=O)CCC(F)CC1C C1(CCC2CCCOC2)C(=O)NCCSC(CCOC)CN1CC=C C1(C(=O)NC(CNC(c2n[nH]c(CC)c2Cl)=O)C)CCC(=O)N(C(C)C)C1 C1(c2n(Cc3occc3)nnn2)(NC2(C3CC3)CC2)CCCN2CCCCC12 Cc1csc(CC(=O)NC2(C3CCCN3C(c3ccns3)=O)CC2)n1 C1(C(=O)NC2CCC(N(C(=O)COCC(F)F)C)CC2)CCn2ncnc2C1 c1(C(=O)NC(C2(O)CCN(C(c3cc(F)cc(F)c3)=O)C2)C)nn(C)c(Cl)c1Cl C(CC(C(=O)NCC1CC1(C)C)NC(=O)CCN(C)C)OC c1(C(=O)NC(CCCNC(C2(OC)CCOC2)=O)C)c(SC)cccc1F N1(C(c2ccc(C(=O)NC(C)C)o2)C(=O)NC)CCC(S(=O)(=O)N(CC)CC)C1 N1(C(=O)CC2(O)CCCC2)CC2CCC(C1)N(C(c1n[nH]cc1Br)=O)C2 C1(CC(=O)NCCC2N(C(C=C(CCC)C)=O)CCOC2)(CF)CC2(CCC2)C1 C(C)(C(C(=O)NCC(C)(C)C(C)(C)O)C(C)C)NC(CCCOCCC)=O N1(C(CNC(c2ccccc2)=O)=O)CCC2CC1CN(C(c1csc(O)n1)=O)C2.C N1(C(COCCCCC)=O)CCC(C)N(C(c2nc(COC)oc2C)=O)CC1 C(=O)(C1CNC(=O)c2ccnn21)NC(C)C(C)(C)NC(=O)C=Cc1cccnc1 CN1C(=O)CCC1C(=O)NCC(C)(F)CNC(=O)CC1CCCCC1O CC1CC(CNC(=O)C=C2CCC2)CN1C(=O)C(Cc1ccccc1)N(C)C C1(CN(C(C2(CCOC)CCC2)=O)C)CCCN1C(c1ccoc1)=O c1(Cn2c(-c3cccnc3O)nc(C(CCC)C)n2)c(Cl)cccc1Cl N1(C(c2c(CC)n(C)cc2)=O)CCN(C(c2cc(O)nc(N(C)C)n2)=O)C2CC12 N1(C(CCC(C)NC(c2cncc(OC)n2)=O)=O)C2C=CCC1CCC2 CCC(C)C(=O)NCC(C)(C)CNC(=O)CNc1cccnc1 C#CCC(C)C(=O)NCC#CCNC(C1(c2ccn(C)n2)CC1)=O C(=O)(CCCS(N)(=O)=O)NC(CCn1cc(C2C(C)CCC2)nn1)C(C)(C)C N1(C(C2C(C)(C)C2)=O)CCCC2CN(C(c3cc[nH]c3C3CC3)=O)CC12 C1(C)(CNC(N2CCCC(CCCC)C2)=O)CCCN(C(=O)OC(C)(C)C)C1 N1(C(C2(CC(C)C)COC2)=O)CCCCC(CNC(=O)C(=O)Nc2ncc[nH]2)C1 N1(C(c2cccc(COC)c2)=O)CCN(C(=O)COCCCC(C)C)C2CC12 O=C(C1=CCS(=O)(=O)C1)NCC1CC1NC(c1cnc2n1CCOC2)=O c1(CN2CC(C)(C(N(Cc3nnc(CC)o3)CC)=O)C2)cc(F)cc(F)c1 c12ccn(n1)C2.c1(COCC(C)OC(C2CC2)=O)ccccc1 c1(CC)cc(C(=O)NCC2CCN(C(=O)CCc3ccn(C)n3)CC2)ccc1O C1(CN(C(=O)C(c2ccc(Br)nc2)(F)F)C)CCCN(C(C2CC2F)=O)C1 C1(COCC)(NC(c2c(C)coc2C)=O)CCN(C(=O)C(F)CC2CC2)CC1 c1(C(=O)N)cc(Cl)c(Cl)s1.C(=O)(CC(=O)NCCOC1CCN(C(C)=O)C1)NC Cc1ncc(C(=O)NCCC(C)N(C(=O)Cc2ccnn2C)C)cc1N c1(C(=O)OCC)cc(OC)cc(OC)c1Cl.c1(C(=O)OCC)cn(C(C)(C)C)nn1 C1(=O)C(C)(F)C(=O)N2CC(CC(F)C(=O)N1)C2.C(C(O)C(C)(C)C)COC C1(OC(C)C)C(c2ccccc2)CCN1C(=O)C(N1CCC(F)C1)=O C1(NC(CCC=C(C)C)=O)CC2CCC(C1)N2Cc1ccc(F)c(C)c1 CC1CN(C(C2CCCCC2)=O)CCCN1C(C1CCCC(=O)CC1)=O N1(C(C(C=C)(F)F)=O)CCC2(C1)CN(C(C1CCCC(CF)C1)=O)C2 C1(NC(c2cc(OCC)n[nH]2)=O)CN(C(C2(OCC)CCC2)=O)CC2(CC2)C1 C1(C(=O)NCCNC(C(C)(C)C)=O)CC(O)CCN1C(=O)C1=NOCC1 N1(C(C(=O)NCC2CCC(C)CC2)=O)CCC(C2Cc3ccccc32)C1 C12(CNC(C(C3CCOC3)OCC)=O)CCC(CC1)N(C(C1CCOC1=O)=O)C2 C12(CC)CCC(C(=O)NCCC3CCCN(C(=O)CC4(C)OCCO4)C3)(CO1)C2 C#CC1CCCN(C(=O)C(CNC(C2CC3(CSC3)C2)=O)OC)CC1 N1(C(CC(CC)C2CC2)=O)CCC2(CC1)CC2CNC(C12CC(CF)(CO1)C2)=O Cc1ccc2cc(CN3CC4CCC(C3)N4C(=O)C(N)=O)c(Cl)nc2c1 N1(C(=O)CC2CCC(O)C2)CCC2CN(c3ccn4nccc4n3)C2C1 c1(CCSC)nc(C2CN(CC(F)F)C2)n(-c2ccccc2C(F)(F)F)n1 c1(SCC(=O)NCC(O)CNC(C2(CCF)COC2)=O)ccccc1Cl Cc1nccc(C(=O)N(CCC(C(C)C)NC(C2C3CCC(F)(F)C23)=O)C)c1C C(=O)(C#CC1CCOC1)NCC1(C(C)(C)O)CN(C(c2nc(OC)c(C)s2)=O)C1 c1(CC)n[nH]c(=NCC2CC(NC(=O)C(C3CCOCC3)F)C2)s1 C(=O)(CCCC(=O)N(C)C)N1CC(C(C(=O)NCCS(CC)(=O)=O)O)C1 Cc1nn(C2CCC2)cc1NC(=O)C(=O)Nc1ccc(CCC(N)=O)cc1 C(C(COC)CC(=O)NCC(=O)NCc1ccc(F)cc1F)OCC C(=O)(CC(C)(C)C(F)(F)F)NC(C(C)NC(CC)=O)(C)C C12(NC(c3c(C)noc3C(C)C)=O)COC(C1)C(NC(C1CC(C)C1)=O)C2 C1(C(=O)NCC(CC)NC(c2cnc(N)cn2)=O)CN(C)CCO1 CN1CCOC(C(N2CC(C)CC2C(=O)NCC2CCC(O)CC2)=O)C1 Cc1ccc(C2(C(=O)NCC3CC(O)CN3C(C3CCS(=O)(=O)N3)=O)CC2)cc1 C(CN=c1[nH]c2cccc(Br)c2o1)C1N(C(C(C)NC(CC)=O)=O)CCCC1 c1(C(C(=O)N(CCNC(C(=O)NC(C)C)=O)C)N(C)C)ccc(Cl)cc1 C1(COC)CC2(CCN2C(C2CCCC(NC(=O)C(F)C3CCC3)C2)=O)C1 N1(C(C(CCC)OCC)=O)CCCCC(N(C)C(c2ccc(C)cc2F)=O)C1 C=CCCCC(C)(C)CNC(=O)CC(CC(C)C)NC(=O)CC1C=CCC1 C(=O)(C1=NOC2(CCOC2)C1)NC(C)CNC(C1(c2ncco2)CCC1)=O CCC(C(=O)NCCN(C(=O)C(n1ccc(C2CC2)n1)C)CC=C(C)C)C(C)C Cc1cc(N)c(C)nc1C(=O)NCCCS(N)(=O)=O.n12cc(nn1)CN(C)CC2 C1(CNC(c2nc(OC)c(C)s2)=O)CC(NC(C2CCCC23CC3)=O)C12CCC2 Cc1cc(C(N2CCC(C)C(CNC(=O)COC3CCC3)C2)=O)c(Cl)cc1N c1(C(=O)NC2(C)CC(NC(c3c(C)cc(Br)o3)=O)C2)c(C)nc(O)nc1C C=CC1(C(=O)NCCCNC(N)=O)CCN(C(=O)NC2CCO2)C1 c1(C(=O)NCC(CNC(c2ccc(O)c(F)c2)=O)CO)cc(Cl)c(F)cc1F Cc1cccc(C(N2CCC(C)C2)=O)c1.n1(NC(CO)C)ccnn1 c1(C(=O)NC2CC(CCNC(Cc3scc(COC)n3)=O)C2)cc2c(s1)CCC2 N1(C(C(CC2CC2)OC)=O)CC(C)(CNC(c2c(F)cccc2Cl)=O)CC1(C)C c1(CN2CC(NC(=O)Nc3ccc(C)cc3)C2)c(F)ccc(Cl)c1F C1(NC(c2cc(CC)n(C)n2)=O)CN(C(=O)Cc2cc(CC)on2)CC2(CC2)C1 C(=O)(C(C)(C)CO)N(CC(CN(C(=O)Cc1ccc(C(C)(C)C)cc1)C)O)C N1(C(C(CCOC)C)=O)CC(F)(F)CC1(C)CNC(=O)C(F)CC1CC1 N1(C(C)C)CCC(N(C)C(C2(C)CCN(C(=O)CN3CCOCC3)C2)=O)CC1 c1(NC(C2CC(NCC3CCN(C)C3)C2)=O)nc2cc(F)ccc2s1 C(=O)(N(OC)C1CCCCC1)C1(C)CN1.C(=O)(C(C)S(C)(=O)=O)OC N1(C(c2cc(OC)no2)=O)CCCC2(CCN(C(C3CCCCNC3=O)=O)C2)C1 c1(C(=O)NC2C(CNC(C(c3ccc(F)cc3)C)=O)C2)ccc(C#N)cc1O c1(C(=O)NCC2CCC(NC(c3ccc(SC)cc3)=O)C2)cc(F)cc(Cl)c1O C1(C)(CNCc2ccc(C)nn2)CCCC(=O)N1.c12cncc(c1)CNC2=O c1(C(N2CC(CC(=O)NCc3ccncc3)OCC2)=O)cn2ccc(Br)cc2n1 CC1(C)CCCCC1CC(=O)NC1(CNC(=O)CCc2ccc(Cl)nc2)CC1 CC(C)CC(C(=O)NCC(C)NC(c1c(F)ccc2[nH]ccc12)=O)C(C)C c1(C(CC)NC(Cn2ccnc2)C(C)C)ccccc1Cl C1(NC(c2c(C)c(O)ccc2)=O)CCC12CCN(C(=O)CC1=NNC(=O)C1)CC2 N1(C(C(C)(C)C(=O)N2CCNCC2)=O)CCC2(CC1)CC2(C)CO c1(C(=O)NC2C(CCC)C2)ccc(CNC(=O)Cc2cnn(C)c2)nc1 CC1(O)CCC(C(=O)NCC(=O)NC2C=CCCC2)CC1 c1(CC)nc(O)c(C(=O)NC2CC2CNC(c2oc(C(F)F)cc2C)=O)cc1C Cn1nccc(C(N2CCOCC2CCNC(c2ccc(F)cn2)=O)=O)c1=O N1(C(C(C)(C)OC)=O)CCC2(CC1)CN(C(C1CC1C1CC(F)(F)C1)=O)CCO2 Cc1nnc2n1CC(C(N1CCC(C)N(C(C34CC(C)(CO3)C4)=O)CC1)=O)CC2 N1(C(=O)CCC2CCCOC2)CCC2(CC1)CN(C(C1(F)CC1)=O)CCO2 N1(C(C=CC)=O)CCCC12CCCN(C(C1CCCN(C(C)C)C1)=O)C2 C(CC(=O)N1CC2CC2(CO)C1)(C(F)(F)F)NC(c1cncc(C2CC2)c1)=O N1(C(c2c(C(C)C)[nH]cc2)=O)CCOC2(C1)CN(C(=O)CN(C)C(=O)C1CC1)C2 C(CCCC)(CC(=O)NCCC1CCOCC1)NC(C(CCC)CC)=O C(=O)(CCC1=NNC(=O)CC1)NCC1(C)CCN(C(c2cc(N)nc(Cl)c2)=O)C1 CC1CCC(C2CCCC2)CN1C(=O)NCc1csc2ccccc12 c1(CC)c(C)cc(NC(c2cnc(O)n(-c3ccccc3)c2=O)C2CC2)cc1C c1(C(N(CCNC(c2c(C)cccc2)=O)C)=O)cnc(NC2CCOC2)nc1O c1(C(=O)NCC2(NC(C3(C)CSC3)=O)CC(OC)C2)coc2cc(C)ccc12 C(N=c1[nH]ccnc1F)C1C(NC(COC)=O)CCCC1.c12c[nH]cc1NC2=O C(=O)(C1COc2ccc(F)cc21)NC1CCC(NC(=O)Cc2cc(CF)on2)C1 Cc1ccc(C(=O)NCCCCC(C)NC(c2cc(Cl)ns2)=O)c([N+](=O)[O-])c1 C1(C(=O)NC(C)C(C)n2cccn2)CCn2c(C(F)(F)F)nnc2C1 C1(CNC(c2cc(C(CC)C)no2)=O)CCN(C(=O)Cc2ccsc2C)CC1C N1(C(Cc2ccc(C)cc2)=O)CCN(C(=O)Cc2csc(S)n2)C(C)C1C c1(-n2cc(CN3CC(NC(c4nc(SC)sc4)=O)(CO)C3)nn2)cc(C)ccc1C N1(C(COCCC(C)C)=O)CC(O)(C2CCN(C(=O)C=CCF)CC2)C1 C(C(C)(C)C(=O)NC1COCC1CNC(C1(C)CCNC1=O)=O)N(C)C CC1(C)CCC(C)(C(=O)NCC2CCN2C(c2ccc3cnnn3c2)=O)CC1 C1(NCc2cccc(C(=O)OC)c2)COC2(CCN(C(=O)C(C)C)CC2)C1 CC(=O)CCCC(=O)NCC1CC(C(F)(F)F)CCN1C(C1COCCO1)=O c1(C(N2CC(C)N(C(C3CNC(=O)N3)=O)CCC2)=O)cc2cc(Cl)c(F)cc2[nH]1 c1(NCC(=C)F)ccc(S(=O)(=O)NC2CCCc3nc(C)sc32)cc1C#N O=C(C1CCCc2ccccc21)NCC1CC1NC(c1cccc2oncc12)=O C(=O)(C1=Cc2cc(C)ccc2OC1)NC(CC)CNC(=O)Cn1ncnn1 C1(CC(=O)NC2CCC(NC(C3(C)ON=C(C)C3)=O)CC2)CCCCC12CC2 c1(C(N(C2CN(C(c3cc(CO)on3)=O)CC2(C)C)C)=O)cc2c(s1)CCC2=O Cc1coc(C)c1C=CC(N1CC(C)(C)CC1CNC(=O)Cc1cnco1)=O c1(C(N(CC(CCC)O)C)=O)nn(CC)cc1I Cc1ccc2nc(C(N3CCOCC(O)C3)=O)[nH]c2c1 c1(OCC(=O)NC(CC)CNC(=O)C(F)(F)c2nc(C)cs2)nn(C)cc1[N+](=O)[O-] C1(NC(c2c(C)ccnn2)=O)CN(C(C2(C)CSC2)=O)CC12CCC2 c1(CN2CC3(CN(C(c4c(C)ccc(F)c4)=O)C3)C2)c[nH]c2ccc(F)cc12 N(C1CCc2ccccc21)C(CC=CCNC(C1(C)N(C)CCC1)=O)=O CCC(CC)CC(=O)NC(CC(F)F)C(=O)NCCCCCOC C1(N(C(c2c(C)ncnc2)=O)C)CCCN(C(C2CC2C2CC2C)=O)CC1 C1(NC(c2nc(CCOCC)oc2)=O)CC2CC1N(C(C1CCS(=O)CC1)=O)C2 C1(CSC2CC3CC(CO)C2C3)C2C3CC4C1C1C2CC3C41.N CC(C)(C)C(O)C(=O)N1CCC(O)(CCNC(=O)CSCc2ccncc2)CC1 Cn1ncc2c(=O)n(CC(=O)NC3(CF)CCN(C(=O)CC4CC4)C3)cnc12 c1(CC)ncoc1C(=O)NC(c1conc1Cn1cc(Cn2ccnc2)nn1)=O O=C(C1=C(Cl)CCOC1)NCC(C1CCC1)NC(c1cc(Br)ccn1)=O C1(C(=O)NCC2CC(NC(CCCCNC(COC)=O)=O)C2)CC2CCC1CC2 c1(OC)cc(C)c(CNCC2CC(F)(F)C23CC3)cn1 c1(C(=O)NCCOCCN(C)C)nnsc1NC(=O)C1CC1 C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(=O)C(C)(F)F CC1(C)CCC(C(=O)NC2CCN(C(=O)CCc3ncc(F)cn3)C2)OC1 c1(C(=O)NC2(CN(C(CC3C(C)CCC3)=O)C)CC2)cncnc1C(C)C C1(NC(c2cn(C(C)C)nc2)=O)CCN(C(c2nc(=O)cc(N)[nH]2)=O)CC1O N1(C(CSC)=O)CCC(CNCCCCNC(c2c[nH]cc(Cl)c2=O)=O)C1(C)C C=CCCCCCNC(C1CCN(C(C2CC(=O)CCO2)=O)C1CC)=O c1(OC)cc(C(N2CC3CC3(C(=O)Nc3cncc(C(F)(F)F)n3)C2)=O)nn1C c1(C(=O)NC2CN(C(C3(C(=O)NC)CC3)=O)CC(O)C2)cc(C)c(Cl)c(C)c1 C(=O)(C1=NOC(C)(C)C1)NC1C(CC)CN(C(c2c(C)coc2C)=O)CC1 C1(C(=O)NC(COCCOC)C)CC2CCCC2N1C(=O)CC1NC(=O)NC1=O N1(C(C2(N(C)C)CCC2)=O)CCN(C(C23CC(c4ccccc4)C2C3)=O)CC1 N1(C(COC(C2CC2c2cc(Cl)sc2Cl)=O)=O)CCC2CCCCCC2C1 C12(CNC(CS(=O)(=O)NCC)=O)CCCC1CCN2C(=O)C(C)=C(C)C CC(C)CC(C(=O)NC1(CO)CN(C(c2nnc(S)n2C)=O)C1)c1ccccc1 N1(C(C(CC)(C)CO)=O)CCC2(C=C(C(=O)NC(C)C(F)(F)F)C2)C1 CCCC(C(O)C(=O)NC1(C)CCCCCCC1)NC(=O)C(=O)N(C)C Cc1cc(C(=O)NC2CC(O)CN(C(c3cccc(F)c3Cl)=O)C2)c(C)cn1 N1(C(C(=O)NCc2cncc(Cl)n2)=O)CCC(CO)(Cc2ccccc2)CC1 C1(O)(C(C)NC(=O)CCc2ccc(N)cn2)CCN(C(=O)Cc2cscn2)CC1 N1(C(C=CC(CC)C)=O)CCOCC1CCNC(c1ccc(C)n1C)=O n1(CC(=O)NCC(C)N(C(c2[nH]cc(C)c2)=O)C)ncc(O)nc1=O CC(CC1CC1)C(=O)NC1(CNC(C2(N3CCOC3=O)CC2)=O)CC1 c1(C(N2CCC(CC)C2CNC(=O)CC23CCCC2C3)=O)ccc(N)c(Cl)n1 C(C)(C(C(=O)NC(CO)CCC1CC1)C(C)C)NC(c1ncnc(C)c1C)=O CC(CCNC(=O)C1CCC(C)(C)c2ccccc21)N=c1ccnc(S(C)(=O)=O)[nH]1 Cc1c(NC(C2CN(C(=O)CCC(C)C)CCC2C(F)(F)F)=O)ncnc1Cl N1(C(C(CO)NC(C(C)CC#N)=O)=O)CC2CSCC2(C)C1 c1(CC)nnc(C)cc1C(N1CC(NC(C)=O)CCC1C)=O Cc1cccc2c1CNC2CNC1CCN(c2cccc(Br)c2)C1=O c1(OC)ccc([N+](=O)[O-])c(CN2CCN(Cc3cc(B(O)O)ccc3Br)CC2)c1 N1(C(C(C)NC)=O)CCC(CNC(=O)CCCn2cc(-c3ccccn3)nn2)C1 C1(CNC(C(CC=C)C)=O)CCN(C(c2ccc(C(F)F)nc2)=O)C1(C)C N1(C(c2nc(COC)sc2)=O)C2CCC1CN(C(=O)C(C)(CO)OC)C2 O=S(=O)(c1cnc(NCC(O)Cn2cccn2)c(Cl)c1)N1CCSC1 N1(C(C(=O)NC(C)C)=O)CCN(C(=O)Cn2nc3c(n2)CCCC3)C2(CC2)C1 N1(C(C2OCCN(C(C(C)(C)CCCF)=O)C2)=O)Cc2cc(O)nnc2C1 c1(C(N2C3CN(C(CCN4C(=O)CCCC4)=O)C(C3)C2)=O)nnn2c1COCC2 C1(C(N2CCC(CCNC(CN(C)C(=O)C3CC3)=O)C2)=O)CC2(CCC2)C1 C(CCCC(C)(C)C(=O)NNC(=O)C(C)NC(N)=O)NC(C1ON=C(CC)C1)=O C1(CC)CN(C(C2CC(=C3CCC3)C2)=O)CC1NC(=O)CC(O)C1CC1 C(=O)(C1CCc2c(Cl)cccc21)N1C2(CNC(CC(CN(C)C)O)=O)CCC1CC2 C1(C(=O)NC2CCN(C(C(C)C)=O)C2Cc2ccccc2)CC12CCCCC2 C1(O)(C(C)NC(c2n(C(C)C)nnc2)=O)CCN(C(C2CCOC(C)C2)=O)C1 C1(CNC(C2ON=C(CC)C2)=O)CC(C)CN(C(c2cc[nH]c2C)=O)C1 c1(C(=O)NCCCN(C(=O)C=C2CCN(C)C2)CC)cn(C)nc1C(C)=O C1(C(N2CC(CNC(CC#N)=O)OCC2)=O)C2CCC(F)(F)C12 C#Cc1ccc(C(N2CCC(CC(=O)NCC(C)(CC)CO)C2(C)C)=O)cn1 C(CCCS(C)(=O)=O)NC(NC(C1CCCOC1c1ccc(Cl)cc1)C)=S C(=O)(C1COc2ccccc21)NCCNS(CCCOC)(=O)=O c1(OC)ccc(C(N2CCC(CN(C(=O)CC3CC3)C)C2)=O)cc1OC1CC1 C(c1ccncn1)=CC(=O)NCCCOCCNC(=O)CC12COC(CF)(C1)C2 C1(N(C(c2[nH]nc(OC)c2Cl)=O)C)CN(C(c2ccoc2Cl)=O)CCC1C C1(C(=O)NC2(C(C)O)CC2)COC(CNC(=O)CCc2cnn(C)c2)C1 N1(C(Cc2cccc(OC)c2)=O)CCC(C2(O)CCN(C(=O)C(C)(C)F)C2)CC1 C(C(CNC(=O)Cc1ccnn1CCF)CO)NC(C1(CS(N)(=O)=O)COC1)=O CC1(C)OC2(C(=O)NCC3CC(NC(c4cc(O)ncn4)=O)C(O)C3)CC1C2 CN1C(=O)CCCC(NC(=O)COC2(C)CN(C(C3CC4(CCO3)CC4)=O)C2)C1 C(=O)(CCC(C)C)NCCN(C(C=CC=CCC)=O)C1CC1 c1(OC)ccccc1S(=O)(=O)NCC1CCN(C(c2cccc(F)c2Cl)=O)C1 c1(C(N2C(C)(CNC(C(CSC)C)=O)CCC2)=O)ccc(Br)c(F)c1F N1(C(C2N(C(C3CCCC(=O)C3)=O)CCN(C)C2)=O)CCC2CCCC2CC1 N1(C(c2c(CC)c[nH]c2)=O)C(CC(=O)NCC2CCC(C(N)=O)O2)C2CCCC12 c1(N2CCN(C(c3c(CC)noc3C)=O)CC2CCO)nc2cccc(C)c2o1 c1(C(N2CC3C(CNC(CCCC(C)=O)=O)(C3)C2)=O)cc2c(s1)COCC2 C(=O)(CCCC(=O)N(C)C)NC1CC(F)(CNC(C(CC)N(CC)CC)=O)C1 N1(C(C2C(OC)CCCC2)=O)CCC(C)N(C(c2cccc(O)c2)=O)CC1 C1(C(=O)NCCC2CCCC3CC23)(CNC(C2CN(C(C)C)C2)=O)CC(C)(C)C1 C(C(C)N=c1nc(O)c(Br)c[nH]1)NC(c1c(C)c2c(s1)cccc2)=O CC1CC(CNC(=O)CC2CC2)CN(C(=O)C(C)(C)CN(C)C)C1 N1(C(CCC2N(C(C)C)CCC2)=O)CCc2n[nH]cc2C1.c12cccc(c1)CN2 c1(C(=O)NC2C(CC(=O)N(C(CC)C)CC)C(O)C2)cc(O)cc(=O)o1 C1(C(N(CCCCCNC(C2CC3CC3C2)=O)C)=O)CCOC(=O)CC1 C(CCCCCC(=O)NC1CCN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1(C)C)SC c1(C(N2C(CNC(C3C4CCC34)=O)CC2)=O)cnc(O)c(C(F)(F)F)c1 c1(C(=O)NCCN(C(C(C)NS(C)(=O)=O)=O)Cc2ccccc2)cnnc(O)c1 c1(N(CCC(=O)CCO)Cc2ccccc2C(=O)O)ccc(Br)c(Cl)c1 Cc1nc(N)cnc1C(=O)NC1CN(C(c2ccc(CCF)cc2)=O)CC12CC2 C(=O)(CC1=CCCC1)N1C(CCNC(C(C)N(C)CC)=O)COCC1 C#CC1(C(N2CC3(CCC3O)C2)=O)CCN(C(=O)C(C)CCC)CC1 C(=O)(C(C1CC1)N(C(=O)C(C)C)C1CC1F)N(CCCC)C(=O)OC(C)(C)C c1(C(=O)NC(C2CCCCN2C(=O)Cn2cnccc2=O)(C)C)cc(Cl)ncc1 O(NC(=O)C(CNC(c1cnn(C)c1)=O)CC(C)C)CC=C N1(C(c2cn(C)nc2)=O)CCC2(CC1)CC(CNC(=O)CSCc1cccs1)C2 N1(C(c2c(CC)oc(C)c2)=O)CC2CCCC1C2CNC(c1cn(C)nc1O)=O N1(C(C(C)(CO)NC(C2COCC2(C)C)=O)=O)CC2(CCOC2)C1 N1(C(c2cccc(N(C)C)c2)=O)CCC2C(C1)CN2C(C1CC2C=CC1C2)=O N1(C(CC=C)=O)C2CCC1CC(F)(CNC(c1cccc3sccc13)=O)C2 Cc1ccnc(C(=O)NC2CC=C(C(=O)NCC3CCC4(CC4)C3)C2)c1N N1(CCNC(C(C)NC(CC)=O)=O)CCC(NC(=O)C(CSC)OC)CC1 C(=O)(CCCCC(F)(F)F)NC(C)Cn1cc(COC(=N)O)nn1 C(=O)(C1=COc2ccccc2O1)N(C1CC(NC(C(CCOC)C)=O)C1)C C(=O)(C(O)CC(C)(C)C)N(C1C=CC(C)(C)CC1)C C1(NC(CC2C(OC)C2)=O)(CO)CCN(C(C2(c3cnccc3C)CC2)=O)CC1 N1(C(=O)Cc2csc(Cl)n2)CCN(C(c2ccc(F)s2)=O)C(CC(F)(F)F)C1 N1(C(CC(C)(C)SC)=O)CC23CCCC2(C1)CN(C(C1CCC12CCC2)=O)C3 c1(C(=O)NC2CC(NC(C3CCC(=O)C3)=O)CC2O)cccc(F)c1Br N1(C(C(N2CC(C)C2)C)=O)CCC(C(N2CC(N(C)C)C(C)C2)=O)C1(C)C N1(C(c2c(OC)ccs2)=O)CCN(C(=O)C=Cc2cncn2C)C(C)CC1C c1(C2(C(=O)NC(C)CNC(c3cccnc3O)=O)CC2)ccc(Cl)cc1Cl Cc1ccc2sc(=NCC34CC(NC(CSCCC5CCCC5C(C)C)=O)(C3)C4)[nH]c2c1 N1(C(C(C(C)C)(C)C)=O)CC(NC(c2cn(CC(N)=O)nn2)=O)C2CCCC2C1 c1(C(=O)NC2CN(C(c3cccc(C#C)c3)=O)CC(C)C2)ccc(C)c(C)c1I C1(CNC(C2C(OC)CC2)=O)CC2CCC1N(C(c1ccc(F)c(C#N)c1)=O)C2 C1(C(=O)OC)(OC)CCN(C(=O)CN2CC3CCC2C3)C1 c1(C(C)CNC(=O)N(CC(F)Cl)C)cnc[nH]1 C1(NC(c2nnnn2C)C)CCN(CC(F)(F)F)C1=O CC1C(NC(=O)COC2(C)CCC2)CCCN1C(=O)CCNc1ccccn1 CC1=CCC(C(=O)NCC2(F)CC(CNC(c3cnoc3C)=O)C2)CC1 C12(CNC(c3ccc(CCC)cc3)=O)CCC1CCN2C(=O)CC(F)F c1(C(=O)NC2CCN(C(c3cc(OCC)ncc3)=O)CC2)ccc(Cl)c(C#N)c1 C1(C(C)C)CCC(C(N2CCC(CC(C)C)C2)=O)N1C(=O)CC1COCCO1 C1(C(=O)NC(CCCC)(C)C)CN(C(C2CCCN2C)=O)CC1(F)F CCCCC(O)C(=O)NCCC1CC(NC(C2(c3ccc(Cl)cc3F)CC2)=O)C1 Cc1oc(C#N)cc1C(N1CC(C(=O)NCC2(C#N)CCC2)CC1(C)C)=O Cn1cnc(S(=O)(=O)N(C2CC2)CC2CCCC(C(F)(F)F)C2)c1 c1(C(=O)NCC(CNC(C(CCOC)C)=O)C)ccc2c(c1)C(=O)CCCC2 N1(C(c2nccc(N(C)C)c2)=O)C2CCC1CN(C(C1CCC(C#N)CC1)=O)C2 C1(C(N2CCC(CC3CC3)C2)=O)CCN(C(=O)c2cccnc2CO)O1 C#Cc1cc(NC(C2CCCN(C(=O)C(C)(C)CCOC)CC2)=O)ccc1C c1(C(=O)NC2CCN(C(CN(C(=O)OC)C)=O)C2C)cc(C)c(C)c(Br)c1 c1(C(C)=O)nc(C(N2CCC2C(=O)N(CCC(C)C)CC23CCC2CC3)=O)cs1 S1(=O)(=O)c2ccc(cc2)N1.Cc1cc(C(N)=O)ncc1NC(=O)C1CC1 C(CCCCN=[N+]=[N-])NC(C1CCCC(NC(CNS(N(C)C)(=O)=O)=O)C1)=O N1(C(CC(=C=C)C)=O)CCC(NC(c2cnn(C(C)C)c2C)=O)C(F)C1 C1(O)(C(=O)NCCC(C)(C)NC(C(CN(CC)CC)F)=O)CN2CCC1CC2 C(=O)(CCCC(C)(C)CC)NC(CCCCn1cc(C(=C)C)nn1)C c1(C(=O)NCC(CO)NC(C(C)OC)=O)cccc(CC#N)c1 N1(C(C(C)OCC)=O)CC2CCN(C(=O)Cn3c(C)csc3=O)C(C2)C1 C(=O)(CC(O)CC(C)C)N1CCCC(C(=O)N(CC(C)C(=O)OC)C)(CC)C1 c1(C(=O)NC(CC)CNC(c2cccnc2C(F)F)=O)cc(C#N)cc(C)n1 c1(C(C)C)scnc1C(N1CC(=C(F)CNC(=O)CC(C)c2cccnc2)C1)=O c1(C(C)NC(c2nnnn2CCCSC)C2(CC)CCC2)ncc(Br)cc1C C1(CCNC(CC2CC(OC)C2)=O)CCCCN1C(C1CC(C)(O)C1)=O n1(CCCC)nnnc1C(C)(CC1CCCCC1)NC(C)Cc1cccs1 C1(F)(C(N2C(CNC(c3ccc(NC(C)=O)s3)=O)CC2)=O)CCCCC1 CC(C)C(O)C(C)(C)C(=O)NCC(C(=O)N1CC(OCC(F)F)C1)N(C)C N1(C(C2(CC)N(C(C(CCC)NC(N)=O)=O)CCC2)=O)CC(=O)N(C)C(C)C1 c1(CC(C)C)nccc(NC(C2CCN(C(C3CNC(=O)C3)=O)C2C)=O)n1 C1(NC(=O)C=CCN2CCOCC2)CC12CCN(C(C1OCCCO1)=O)CC2 C1(N(C)C)CCC(C(=O)NCCC2CC(NC(c3cc(Cl)n[nH]3)=O)C2)CC1 Cc1oc(C(F)(F)F)nc1C(=O)N(C)CCOCCNC(c1cn(C)nc1O)=O c1(NC(=O)NCCC2CCCC(C)C2)ccc2c(c1)C(O)CC2(C)C C1(OC)CCC(c2nc(-c3cccc(N)n3)nn2-c2nc(Br)nn2C)CC1 C1(NC(Cc2c(SC)cccc2)=O)COC2(C1)CN(C(=O)CCC(=O)OC)C2 c1(CC(=O)NC(C#C)C(C)C)ccc(OC)c2ccccc12 C1(NCc2nc(CCC)on2)CCN(C(=O)CCn2ccnc2)CC1C C1(C(=O)NCC2(CCC)CCC2)CCCN(C(=O)Cc2cc(C)n(C)n2)C1 N1(CC(=O)N(CCCCN(C)C(c2cc(Cl)ns2)=O)C)CCCCS1(=O)=O C1(C(=O)NCC2C=CC(NC(C3C(C)CC(=O)N3)=O)C2)Cc2cncn2C(=O)N1 c1(OC)cc(CN)ccc1-n1ccnc1.C1(C(N2CCOCC2)=O)(CN)CC2(CC2)C1 C1(C(N(CC(O)CN(C)C(C2CCCCC2)=O)C)=O)(CO)CCCCC1 N1(C(CC2(C=C)CC2)=O)CC2CC(NC(=O)C(C)NC(=O)C(C)(C)C)C1C2 CN1C(=O)CCCC1C(N1CCC(C)(C)C1C(=O)Nc1cccc(CO)c1)=O C12(OCC)CCC(C(=O)NC3CC3CNC(c3sncc3C)=O)(CC1)C2 C1(NC(c2cnc(OC3CCOC3)cn2)=O)CC12CC(Cc1ccccc1)C2 n1(CC)cnc2c(NC3CCCCCN(C(=O)C4=CCCS4)C3)ncnc12 C12(CNC(=O)OC(C)(C)C)CC(NC(=O)C(C)CN3CCOCC3)(C1)C2 C1(C2(C)CC2)COCCN1C(=O)CC1CCCN1C(C1COCCO1)=O C(=O)(CCCCCCCCC(=O)N1CCCCC2(CCN(C3CC3)C2)C1)OC C1(NC(COC(C)=O)=O)CCC2(C1)CN(C(C1CNC(=O)C1)=O)C2 C(=O)(N=c1[nH]nc(Cc2ccnc(OC)c2)s1)NC1C(CCC)CCC1 C1(C)(C(N2CC(CNC(c3c(C)ncc(Cl)c3)=O)C2)=O)COC2COCC12 Cc1cccn2c(C(N3CC(CNC(c4ccc(O)nc4)=O)C(O)C3)=O)cnc12 c12ccc(cc1F)c1ccc(cc1)[nH]c2=O.Cc1cc(OCC2CCOC2)no1 Cc1cc(C(=O)NCC23CC2CN(C(C2(C(N)=O)CC2)=O)C3)nc(C)n1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC(NC(=O)C(F)C(F)(F)F)C2(CCC2)C1 C(C)(CCCCNC(=O)Cc1nc(-c2cccs2)oc1C)NC(COCC)=O c1(C(=O)NCC(=CC(=O)N(CC(=C)C)C)C)cnnn1CC C1(N(C)C)(CO)CCN(C(C2CCC(=O)N(Cc3ccccc3)C2)=O)CC1 N1(C(C2CCCC(C(N)=O)C2)=O)CCC(CN(C(=O)COC2CC2)C(C)C)CC1 N1(C(C2(C)COCCO2)=O)CCC(NC(c2ccc(Cl)s2)=O)C(CO)C1 C1(NC(c2c(C)cn(C(C)C)c2)=O)CC(NC(=O)CN2CC=CC2)C12CCC2 Cc1cccc2c1OCC2C(=O)N1C2CCCC1CN(C(c1[nH]nnc1C)=O)C2 N1(C(C2C(C(C)C)C2)=O)CCCC2C(NC(C3CC(C)(C)CCO3)=O)C(C)(C)C12 c1(C(C(=O)N(C)CC2N(C(CC=CCCCCC)=O)CCC2)C)cccc(F)c1 c1(CC)noc(C(N2CCC(CCNC(=O)Cc3cccnc3)C2)=O)c1C c1(NC(c2cc(OC)c(C)c(OC)c2)=O)[nH]c2ccccc2c1C c1(C(N2CCCN(C(CC(=C=C)C)=O)CC2)=O)ccc2n[nH]c(C)c2c1 C=CCCC(C(=O)NC1CC(N(C)C)C1)NC(C1CCCCO1)=O C#Cc1cc(C(N2CCC(C)(CCNC(=O)COC3CC3)C2)=O)cc(Br)c1 N1(C(CCC#N)=O)CC2CCC(NC(C3CC4CCC(C3)C4O)=O)(C2)C1 C1(CC(=O)NC(C23CC(CCO2)C3)C)(OC)CCN(C(c2ccon2)=O)C1 C1(NC(C(CCC)O)=O)CN(C(C2CCC(C(C)(C)C)O2)=O)CC2(CC2)C1 CN=c1[nH]nc(CC(=O)NCc2cn(CC(N3CCCC(NC(N)=O)C3)=O)nn2)s1 Cc1ccc(NC(=O)C(C)(C)CN2CCN(C)CC2)cc1Cl C1(CC=C)(NC(c2ccc(CCC)cc2)=O)CCN(C(c2csc(C)n2)=O)C1 C1(NC(C(C)N2CCCC2)=O)CC2CCC(C1)N2C(=O)CCC1CC(C)(C)CO1 C1(C(=O)NC2CCN(C(C(C)CSC(F)(F)F)=O)CC2)CCc2nn[nH]c2C1 C1(O)(CCNC(CC(=O)OC)=O)CCCN(C(c2cccc(=O)n2O)=O)C1 C12(CC)CCC(C(N3CC4(CCN(C(C5(C)CCOC5C)=O)C4)C3)=O)(CC1)CO2 C1(NC(C2C(CC)CCC2)=O)CCC(CNC(c2ccc(C3CC3)nc2)=O)CC1 N1(C(c2cncc(NCC)c2)=O)CC(O)C(O)C1CNC(c1nnccc1C)=O c1(C(=O)NC(C)C(=O)NCc2ccc(C#N)o2)ccc(C(N)=O)cc1 C#Cc1c[nH]nc1C(=O)NCCN(C)C(c1cccnc1O)=O CCC(C)(CNC(c1ccc(CF)cc1)=O)C(=O)N1CC(C)C(F)(F)C1 c1(C(=O)NC2CC(CNC(c3n(CC=C)ccc3)=O)C2)cccc(C)c1O Cc1onc(C(F)(F)F)c1C(=O)NCC1(O)CCN(C(=O)C(O)CCN(C)C)C1 N1(C(c2c(C)occ2)=O)CCC(NC(=O)CC2CC3(CC3)C2)C1C CC1CCCc2cc(C(N3CCC4(C3)CC4(F)F)=O)nn21 Cc1cc(CCC(=O)NCC2CN(C(c3ccnn3CC3CC3)=O)C2)cc(F)c1 C(=O)(CCCN=[N+]=[N-])N1CC(O)(CN(C(CN(C(=O)OC)C)=O)C)C1 N1(C(CCN(c2ccc(Cl)cc2)C)=O)CC(NC(=O)CCN2CCC2)C(C)(C)C1 C1(CNC(c2cn(C)nc2C(C)C)c2n(C(CC)(C)C)nnn2)CCC(=O)NC1 C1(CC)CN(C(=O)C=C(C)CNC(=O)C(C)CC#N)C1(C)C.C(=O)(N)OC N1(C(C(CC)C)=O)CC2(CCCC(CNC(C3CCC(=O)N3C)=O)O2)C1 N1(C(C(CCC)OC)=O)CCN(C)CC1C(=O)NCC1CC(=O)NC1=O c1(C(=O)NCC2CCN(C(CC3CC(OC)C3)=O)C(C)C2)nccc2nn[nH]c12 c1(C(=O)NC2CCCC(NC(c3cc(OC)n[nH]3)=O)CC2)cccc2ncsc12 C1(NC(=O)CCc2nc[nH]n2)CC2CC(NC(=O)COc3ccc(F)cn3)C2C1 N1(C(C(C=CC)O)=O)CCCN(CCCCNC(c2cccc(CC)c2)=O)CC1 CC1CCC(NC(c2ccc(CNC(C3C4COCC34)=O)s2)=O)C1 N1(C(c2cc(C(C)=O)on2)=O)CCC(C(F)F)(CNC(=O)C(C)(C)CF)C1 N1(CCCc2ccc(C)cc2C)CC2CC1CC2(C)O C(C(C)(CC(C)C)NC(=O)CC1CC2CCC1O2)NC(c1c(C)nc(CC)s1)=O c1(CC(=O)NC(CNC(C2N(CCC(C)C)CCC2)=O)(C)C2CC2)ccnc(O)c1 C1(CNC(CN(C(c2n(CC)ccc2)=O)C2CC2)=O)CCC(=O)NC1C CCC(C)(CO)C(=O)NCC1(NC(c2cc(=O)c(Br)c[nH]2)=O)CCOC1 CC1CC(NC(c2ccsc2)=O)CN1C(C1CCOC(C)C1)=O c1(C(=O)NCCC(C)NC(c2n(CC)ncc2)=O)ccnc(C(N)=O)c1 c1(C(=O)NC(C2CCCC2)CNC(C2C(OC)C2C)=O)cnc(OC)c(Cl)c1 N1(C(C=CC(CC)=CC)=O)CCC(O)(C(C)NC(=O)CCSCCCC)C1 C1(NC(CCOCC)=O)CCN(C(c2sc(CC(F)(F)F)nc2C)=O)CC1C c1(C(N2CC(C)OCC2)=O)cn2c(n1)CCN(Cc1cc(Br)co1)CC2 c1(CC(=O)NC2CC3CN(C(c4c(C)snc4)=O)C2C3)cccc2c1SCCC2 C(=O)(CC(C)(C)CC(F)F)N(CCC(C(C)C)NC(=O)C=CC1CCOCC1)C c1(SC)cc(C(=O)NCC2C3CN(C(=O)COCP(C)(C)=O)CC23)c(C)o1 N1(C(c2c(CC)ncs2)=O)CCCC(COC)(NC(=O)C(C)c2ncco2)C1 c1(C(=O)NCC(CC)NC(=O)CC2CCC(C)(O)CC2)c[nH]nc1S(N)(=O)=O C1(CNC(C2CC(C)(CC(C)C)C2)=O)CCCCN1C(c1cc(O)n(C)n1)=O N1(C(C(C)SC)=O)CCCCC1.C(CC(C)NC(=O)COC)N(C)C N1(C(C2CC=C(C)CC2)=O)CC(NC(=O)Cc2cnsc2)C(C2CC2)C1 Nc1c(C(=O)N(C2(c3cn(C4CCC4)nn3)CC2)CCO)cnn1CCO CCCCCC(C)(C)C(=O)N1C(C(=O)NCCF)CC2CC12 N1(C(c2ncn(C)n2)=O)CCCC(F)(CNC(c2ccc(C(N)=O)nc2)=O)C1 c1(-c2cnc(=NC)[nH]c2)cnc2[nH]cc(C(=O)NCc3cncc(C)c3)c2c1 C1(NC(C)=O)CCC(C(=O)NC(C)CCNC(=O)COc2cncc(C)n2)CC1 N1(C(C2(C)CCCOC2)=O)CCOC(C(N2CCOC(CF)C2)=O)CC1 C1(CC(=O)OC)C(=O)NCCN1C(c1c[nH]cc(C)c1=O)=O N1(C(c2on(C)c(=O)c2)=O)CCOC2CCN(C(C3CCCS3(=O)=O)=O)CC12 C1(NC(=O)CN(C(=O)C=Cc2ccc[nH]2)C2CC2)CCOCC1F CC(C)CCC(C)NC(=O)CC1CCCN1C(c1cn[nH]c1)=O C12(CC(=O)NC(CC#C)(C)C)CCC1CN(C(c1cccc(C3CC3)n1)=O)C2 c1(CNC(C2CCCCCC2)CO)cccc(F)c1Cl c1(C(=O)NCC2(C(N(CCN(CC=C)C)CC)=O)CC=CC2)cncc(O)c1 C1(CNC(CSC)=O)CC2(CCN(C(C3CN(C)C3)=O)CC2)CO1 N1(SCC)CCC(N=c2nc(NC3COC4(CCC4)C3)c3c([nH]2)c(C)nn3C)CC1 c1(C(=O)NCCC2CCCN(C(c3nccc(C)c3)=O)C2)c[nH]c(=N)nc1C Cc1ccc2c(c1)C(NS(=O)(=O)c1ccc(I)cc1)CC2(C)C C1(O)(CNC(Cc2cc(C)sc2)=O)CCCN(C(C2(C#N)CCCCC2)=O)CC1 CN=c1ccc(C(=O)NC2CCC(CNC(=O)CCOCCN(C)C)CC2)c[nH]1 c1(C(=O)NC(C(=O)N2CC(=O)O2)C)ccn(C)c1.C#CCOC c1(CN2C(C(=O)N(CCCCO)CC)CC(=C)C2)ccc(Br)nc1F c1(OC)ccc2c(C(N3CCC(NC(C4CCCC(C)(C)C4)=O)C3)=O)cnn2c1 C1(c2c(C)n(C)nc2)CCCN1N1CCC(COC(F)F)CC1 CC(F)(F)C(F)(F)CC(=O)N1CC=CC(NC(c2cc(Cl)sc2Cl)=O)C1 C(=O)(C(C)CC(N)=O)NC1CC(NC(CCc2onc(CSC)n2)=O)C1 c1(CC(=O)NC2CC(CNC(=O)C=CC3CCCCC3)C2)cccc(Cl)c1F N1(C(C(C(C)OC)O)=O)CCn2ncc(CN(C(=O)Cc3cnc(C)s3)C)c2C1 Nc1cc(F)cnc1C(N1CC=C(C(=O)NCc2ncc(F)cn2)C1)=O CCC(CC)C(C)C(=O)N1CCC(NC(c2cc(N)c(C)c(N)c2)=O)C(C)C1 N1(C(C23N(C(C(CCC)OCC)=O)CC(C2)C3)=O)CCCC2(CCOC2)C1 C1(NC(c2cnn(CC)c2C)=O)CN(C(c2cccc(Cl)c2N)=O)CC(C)(C)C1 N1(C(c2c(C)oc(Cl)n2)=O)CCCC(C2CCN(C(c3nnsc3C)=O)CC2)C1 N1(C(C(=O)NCCCF)=O)CCc2c([nH]c3ccc(F)cc23)C1 C1(CNC(CCCOC(C)C)=O)CCN(C(C2CN(C(C)C)C2)=O)C1(C)C C1(NC(c2scc(CNC(C(CC)C#N)=O)c2)=O)CCOC(C)(C)C1 C1(O)(CNC(COCC)=O)CCCN(C(=O)C(c2ccncc2C)C)C1 c1(C(=O)OC)cc(C)n(-c2ccc(C(C)NCC(C)Oc3ccccc3)cc2)n1 Cc1ccccc1CC(=O)NCC(C1CCCN1C(=O)C(C)C#N)(C)C c1(NC(=O)NCC(c2ccc(Cl)cc2)=O)cc2c(nc1O)CCSC2 C1(C(=O)NC(c2snnc2C)CC)(NC(c2ccccn2)=O)CC(F)(F)C1 C(c1ccc(-c2ccccc2F)s1)=CC(=O)NC(C(C)NC(=O)CNC=O)CO c1(C(N2CCCC23CCS(=O)(=O)C3)=O)ccc(Cc2cccs2)c2c1CNCC2 C(Cc1cnc[nH]1)(C(=O)NCCCO)NC(C(c1ccoc1)OCC)=O C1(C(=O)NCCO)C2CCC(=O)C12.CC(C)COCCCNC(c1ccns1)=O C=CC1(CC(=O)NCCCn2cccn2)CN(C(=O)CC2(C)OCCO2)C1 O=C1NC2(CNCC3(c4ccccc4)CNC(=O)C3)COCC2O1 c1(CN(c2cc(C)[nH]n2)C(C)(CCI)c2n(CCCOC)nnn2)ccc(Cl)cc1 c1(C(N2CC3N(C(CCCC(N)=O)=O)C(CC3)C2)=O)cc2n(c1)CCS(=O)(=O)C2 CCC(C)C(C)(O)CNC(C1CCCC(NC(=O)C(O)CC(N)=O)C1)=O Cc1cc(N)c(C(N2CC3(CCN(C(C4(n5ccnn5)CC4)=O)C3)C2)=O)cc1F N1(C(c2cc(C(C)(C)C)[nH]n2)=O)CCOC(CNC(=O)CCC2CCC2)C1 c1(C(C)C)cc(C(N2CCC(N(C(=O)CSc3ccncc3)C)CC2)=O)n(C)n1 c1(CC)noc(C)c1CC(=O)NC1CCC(C)(CNC(C23CC(C)(C2)C3)=O)C1 C1(C(N2CCC(CNC(c3n(COC)ncc3)=O)CC2)=O)CCOC(=O)CC1 C12(C(N(C)Cc3cccs3)=O)CCN(C(=O)Cc3cccnc3)CCC1C2 N1(C(c2c(Cl)cnc(C)n2)=O)CC(NC(c2cc(CF)on2)=O)C(N=[N+]=[N-])C1 N1(C(CC(C)OC)=O)CCOCC1CC(=O)NCC1CC(=O)N(C)C1 C1(C(N2CCC(C(C)NC(c3c(C)cno3)=O)C2)=O)CCc2ncnc(C)c2C1 N1(C(c2c(C)nc(C(C)C)o2)=O)CC2(NC(=O)C(CC(C)C)N(C)C)CCC1C2 C12(COC)CCC(C(=O)N(C(C)CN(C)C)C)(CO1)C2 c1(OC)cc(CC(=O)OC2CN(C(=O)CCCC3CC3)CC2C)c(F)cc1O Cc1nc(O)[nH]c1C(=O)N(C)CC1CCCN1C(C1CCOC1C1CC1)=O c1(C(N2C(CNC(c3ncccn3)=O)CCC2)=O)snc2ccc(Br)cc12 C1(C(=O)NCC2C(NC(C3(C)CC3)=O)CCC2)CCC2(C1)CC2(F)F c1(OC)cc(C(=O)NCC2CC(F)(CNC(C3CC34CCOC4)=O)C2)c(F)cn1 c1(NCC)cc(Cl)ccc1C(N1CC(NC(c2cccc(C)c2)=O)CC1CO)=O S(=O)(=O)(CC(=O)N1CC(N(C(=O)CN(C2CCC2)C)CC)C1)NCC C1(O)(CCNC(C2(CC#C)CCCOC2)=O)CCN(C(=O)Cc2ccon2)CC1 C(c1cccc(Cl)c1)=C(C(=O)NC1CN(C(C(CC#C)O)=O)CC1C(F)(F)F)C N1(C(Cc2n(C)ccn2)=O)CC(NC(=O)Cc2ccco2)CCC(O)C1 c12cc(cc3c1OC(C)C3)O2.CCC(C)C(=O)N1CC(CN)C1 c1(OCC)ccc(Cl)c(C(N2CC(NC(=O)CCC(CC)SC)CC(C)C2)=O)n1 c1(CC)cc(C(=O)NCC2CCCN2C(c2cc(COC)no2)=O)sc1Br C1(CNC(=O)Cc2ccc(OCC(F)F)cc2)C2CN(C(C3CC3F)=O)CC12 C=C1CC(C(=O)NCC(c2ccncc2)(C)O)N(C(c2ccoc2CC)=O)C1 CCC(=O)C(=O)N1CC(n2cc(CNC(c3c(CSC4CC4)ocn3)=O)nn2)C1 c1(CC(=O)N(CC(F)Cl)CC)ccc2c(c1)OC(F)(F)O2 C1(CNC(COCCC=C)=O)(CO)CCOC1.C(=O)(C(CN(C)C)N(C)C)N N1(C(c2cncc(OCC)c2C)=O)CCOC2(CCC(C#N)CC2)C1 CN(C)S(=O)(=O)N1CC(C(=O)NCCC2(O)CN(C(C3CCCS3(=O)=O)=O)C2)C1 CC1CCCC=C1C(=O)NC(CN=[N+]=[N-])C(=O)NC1CCC(C(N)=O)C1 C(C(C)N=c1ccnc(Cl)[nH]1)NC(C(CCC)CC1CCCCC1)=O CS(=O)(=NC(=O)C(F)c1ccccc1F)N1CCCNCC1 N1(C(c2cccc(NC(=O)OCC)c2)=O)CC2CCN(C(C)=O)CC12 CCCC(CC1CCCC1)C(=O)NCC1C2CN(C(=O)COCC)CC12 c1(N2C(C)C(NC(=O)CCc3cccc(F)c3)CC2)ncc(C#N)c2ccsc12 c1(CC(N2CCC(N(C(=O)Cc3ccnc(Br)c3)CC)C2)=O)cc(F)ccc1O C(=O)(C1CCCn2c(C)nnc21)N(C(C)CNC(c1ccc(CO)nc1)=O)CC N1(C(C23CC(C)(C2)C3)=O)CC2(C=C(C(=O)N3CCC(O)C(F)(F)C3)CO2)C1 C=CC1(C(=O)NC2CC(O)CN(C(=O)Cn3ncccc3=O)C2)CCCCC1 n1(CC)ccc(C(=O)NCC2CCN(C(c3ccns3)=O)C23CC3)cc1=O C=CC1(C(N2CC(NC(c3cc(C)nnc3O)=O)C(C)C2)=O)CCCCC1 C1(CNC(C2=C(C)OCC2)=O)CC2(CCN(C(C34CC(OCO)C3C4)=O)CC2)CO1.C(C)=O C1(C(N2CC(C(C(=O)NC(C(CC)C)C)O)C2)=O)CN(C)C(=O)N1 N1(C(C(CSC)(C)NC(=O)C(O)C2CCC2)=O)CC(=O)NC(=O)C1C N1(C(c2n(C(C)C)ccc2)=O)CC(CNC(c2c[nH]nc2[N+](=O)[O-])=O)CC1(C)C C1(CNC(c2c(C)ccnc2C)=O)CCCCN(C(=O)C2=COCCC2)CC1 c1(NC(C2CCN(Cc3cnc(Cl)c(F)c3)CC2)=O)cc([N+](=O)[O-])ccc1Cl C(=O)(C(C)(C)S(C)(=O)=O)NC1CC(CNC(C(C(C)C)N2CCCCC2)=O)C1 CCC(CC(=O)NC(C(=O)NCc1nnnn1C)C(C)(C)O)CC(C)C N1(C(C(CC)N(C(=O)CCn2cccn2)C)=O)CCCC(C#N)C1 CN(CCc1ccc(Br)cc1)N1CC(C)(C)C(C(c2ccccc2)=O)C1 c1(OC)cc(F)c(C(=O)O)cc1S(=O)(=O)NCc1cc(O)ccc1Cl c1(N2C(CNC(C3CCCC(F)C3)=O)CCCC2)ncnc2[nH]cnc12 CCCC(C)CCCC(=O)N(C)CCN(C)C(c1cc2cccnn2n1)=O C#Cc1cccc(C(=O)NCC(C2CCC2)NC(c2ccnc(C)c2)=O)c1F C(=O)(C1=CCCN(CCO)C1)N(C(=O)C(Cl)(Cl)Cl)C(c1cc(Cl)c(O)cc1F)=O Cc1nc(CC(C)C)c(C(=O)N(CC(=O)O)Cc2nnn(C)n2)s1.c12cn(nn1)C2 C1(N(C(=O)NC(=O)NC2(CCCC)C(C=C)CC2)C)CCOC(C)(C)C1 N1(C(C2CC3(CN(C(c4ccc5cc[nH]c5n4)=O)C3)C2)=O)CCN2CC(O)CC2C1 C(CCCC(=O)NC1CCCC(CNC(=O)C(F)(F)CO)C1)N(C(C)C)C c1(C(=O)NCCCCN(C(=O)CC2CNC(=O)C2)C)ccc(C#N)cc1F C1(CC(=O)NCCCC2CN(C(C3CCO3)=O)CCO2)COCCOC1 CC1CCC(C(=O)NCC2(C3CCC3)CC2)N1C(=O)C(O)CN(C)C N1(C(C(C)N(C)C)=O)CCC(NC(C2(NC(C)=O)CCCCC2)=O)C(C)C1 c1(C(=O)NC2CC(NC(C34CCCCC3C4)=O)C2)ccnc2[nH]nnc12 CCC(Cc1ccccc1)C(=O)NC1CCC(NC(c2n[nH]c(C)c2F)=O)C1 C(CCC(C)NC(C1CCC(C)C1)=O)NC(C(C)OCC(C)C)=O C1(NC(C(COCC)(C)C)=O)CCN(c2ncc(O)cn2)CC(C)(C)C1 CN1CCN(CCNC(=O)NCCC2CCCO2)CC1 C1(C(N(C)CC2CCCS2)=O)CC12CCN(C(c1ccc(O)cc1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NC1CC(CC(=O)N(CCCCC)CCO)C1(C)C Cc1ncc(F)c(=NCc2cc(S(C)(=O)=O)co2)[nH]1 O(S(=O)(=O)CCc1cccc(C(F)F)c1)c1n(C)ncc1 C(CCN=C(NCCN(S(C)(=O)=O)C)NCc1cccc(C2CC2)c1F)OC N1(C(C(CC)CC(C)C)=O)CCC2(CC1)CN(C(c1ccc(Cl)cc1O)=O)C2 C1(NC(c2ccc(SC)o2)=O)C2CC(CN(C(c3cc(C)n(C)c3)=O)C2)C1CO c1(CN2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)C2)ccncc1F C1(C(=O)NC(CCNC(C(C=C)(C)C)=O)C(C)C)C2Cc3ccccc3C12 C12(C(N(c3cccc(Cl)c3)C)=O)C(NC(C3CC4(CC4)CO3)=O)C3CC1C2C3 C1(NC(CCN(C(C)C)C(c2c[nH]nc2Cl)=O)=O)CCCCC1C n1(CCOC)cc(C(=O)NC2CCCC2NC(c2coc(C(F)(F)F)c2)=O)nn1 C1(OC)(CNC(C2(Cl)CCC2)=O)CCN(C(=O)C(O)c2cnc[nH]2)C1 N1(C(c2cccc(C)c2F)=O)C(CNC(=O)C(C)CC2CCCO2)CC2COCC12 C1(C(=O)NCCn2c(C(=O)OC)ccc2)OCCCC1(C)C.C1CCNC(=O)N1C C(=O)(N=c1ccn(CCCO)[nH]1)c1c(CNC(C(CC)NC(N)=O)=O)ccs1 N1(C(C=C(C)Cl)=O)CC2CC(C1)CN(C(=O)Cc1csc3ccc(Cl)cc13)C2 C1(NC(CCC(C)=O)=O)CCCCCCC1NC(=O)C(C)C1CCCO1 c1(C(=O)NC2CCC(NC(C(C)(F)F)=O)C2)ccc(C2(C)CC2(F)F)cc1 C#Cc1ccc(C(=O)NC2CC2CNC(c2cc(C3CCCC3)[nH]n2)=O)cc1Cl c1(C(=O)NC2C(NC(Cc3c(C)ccnc3)=O)CC2)nc(Br)cnc1N c1(CC)ccc(C(C)C(=O)NCCN(C(=O)C(C)(COC)OC)C2CC2)cc1 CC(C)(CCNC(C1CC(CC2CC2)C1)=O)NC(=O)C(CO)c1ccccc1 n1(CC)cc(Cl)c(C(N2CCC(C)(NC(=O)CN3CCC3C)C2)=O)n1 N1(C(C2(C=C)CCC2)=O)CCCC(C(=O)N(CCCC)CC(C)C)C1 C1(NC(c2cn(CC)nn2)=O)CCCC(C(N2CCC(OCCN(C)C)C2)=O)C1 C=CC(C)(O)CC(=O)NC(C1CCN(C(=O)C(c2ccc(C)cc2)C)CC1)C N1(C(C(C)(C)O)=O)CCOCC1CC(=O)NCc1cncc(Cl)c1 Nc1cc(C(N2CC(CNC(=O)CC3CC4(CC4)C3)C2)=O)cnc1Cl CC1(OCC(=O)NC2CCC(NC(c3cnc(N(C)C)o3)=O)C2)CCCC1 N1(C(C(=O)NCc2ncc(-c3c(C)n[nH]c3C)o2)=O)CCC(O)(C2CC2)C1 C1(C(C)NC(C(C)OC)=O)CCN(C(C2(C3CC3)CCC2)=O)CC1 c1(C(=O)NCC2(NC(C(C(CC)C)O)=O)CCC2)cn(C)c(=O)nc1O c1(C2(CNC(C(CC)c3ccccc3)=O)CCC2)ccccc1C C1(CCCO)CN(C(C2C(C(C)(C)C)C2)=O)CCN1C(=O)CN1CCCCC1 N1(C(C2CC23CCCC3)=O)CCC2(CCC2)C(CNC(C2(CCF)CC2)=O)C1 C1(CNC(CC(C=C)C)=O)CCC(C)N(C(=O)CC2CN3CCC2CC3)C1 c1(C(=O)NCC2CC2CNC(C2C3CCC2CC3)=O)cc2ccccc2cc1Cl Cc1cc(C(N2CCCC2(C)CNC(C23CC(C(=O)OC)(C2)C3)=O)=O)nc(O)n1 N1(C(c2cc(OC)nc(OC)c2)=O)CC2CCC1CN2Cc1ccc(O)c(Cl)c1 C1(NC(Cc2c(C)nn(C)c2C)=O)CCCC12CN(C(c1sccc1Cl)=O)C2 C1(NC(C=NOC)=O)CCC2(CC1)CC2C(N1CCOCC1)=O.C1(=O)C(C)N1 Cc1cc(P(C)(C)=O)oc1C(=O)NC1CCN(C(=O)C(O)C(C)C)CC12CCC2 C(=O)(C1=C(Cl)CCOC1)NC1CC(C)CN(C(=O)Cc2cnccn2)C1 N1(C(C(COC(C)=O)C)=O)CC=CC(NC(c2nc(C(C)C)oc2C)=O)C1 C(=O)(C(CC)C(F)(F)F)NCC1(CNC(CC=CCC)=O)CC12CCC2 C1(NC(c2c(C)n(C)nc2)=O)CC2CCC(C1)N2C(c1cc2cccn2cn1)=O c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(CO)c1 N1(C(c2n(CCC)ncc2)C(=O)NC2CCC2)CCCC1(C)c1ccccc1 N12CCCC1C2.C1(NC(C(=O)NC2CC2)=O)CCCC1N1CCOCC1 N1(C(C2CCC(=O)N2)=O)CCCCC12CC(NC(=O)CCc1ccccc1F)C2 C1(C(=O)NC2C(NC(c3c(CC)con3)=O)CCOC2)CCCCC1(C)C c1(C(=O)NCC(C=C)C)cc(Cl)ccc1N N1(C(c2cc(C)sn2)=O)CC2CN(C(=O)CC(O)C(C)C)CC(C1)O2 C(=O)(N1CCCc2nccn21)c1c(C)[nH]cc1.c12ncccc1C(=O)NC2 N1(C(CC(CC(C)C)O)=O)CCC2CCN(C(C3CCCCO3)=O)C2C1 N(C1CCCc2ccccc21)(C(C(=O)NCC1C(SC)COC1)=O)CC(C)C Cc1cc2ccc(C(N3CCC4C(NC(C5(C)CC5(F)F)=O)CC34)=O)cn2c1 C(=O)(C(C1CCOC1)SC)N(CC(=O)N(CCO)C(C)C)CCOC c1(C(N2CC(CC)N(C(C3CC(C(C)C)C3)=O)CC2)=O)cccc2cnsc12 C(C(CC(=O)N1C2CCC(C2)C1CNC(C1(O)COC1)=O)C(F)F)N(C)C c1(C(N(C(CC)C(=O)N2CC(NC(=O)COC)C2)C)=O)cnc2[nH]ncc2c1 CC(C)C(O)C(C)C(=O)N(C)CC1CCN(C(c2nccc3occc23)=O)C1 C(C)(CCCOC(C)C)(c1n(CC=C)nnn1)NCC(C)(C)C1(O)CCC1 C1(CCNC(=O)CN2CCSCC2)CN(C(C2CC2(Cl)Cl)=O)CCCO1 C(=O)(CC(C)C(F)F)NCCC1CC(NC(C(C)NC(c2ccccc2)=O)=O)C1 CC(C)C(CN=c1[nH]c(N2CC3CC3(CO)C2)nc2cc[nH]c12)N(C)C c1(OC)ccc(C(C)CC(=O)NC(C)CNC(=O)Cn2nnc(C3CC3)n2)cc1 C1(NC(C#CC(C)(C)C)=O)CCCC2CN(C(C3(C)CCCC3)=O)CC12 c1(C(=O)NC(C(C)C)(C)CNC(=O)CC(C)(C)C)cnc(O)c2cnccc12 C1(NC(C2CCCCN2Cc2ccccc2)=O)C(O)C2CCOC12 c1(C(=O)NC(CC)CC)nc(CNC(=O)C(F)C2CCCC2)oc1C C1(C(=O)NCC2(CNC(C(C)OC3CCCC3)=O)CCCC2)CCC(F)CC1 C1(NC(C(CC(C)C)C)=O)CCSC12CN(C(C1(O)CC(CF)C1)=O)C2 c1(C(=O)NCC#CCNC(c2cn(CC)nc2C)=O)cc(F)cc2cccnc12 c1(C(N2CCC(NC(C3C(C)=CCS3)=O)(CF)C2)=O)c(O)cccc1F Cc1ccc(C(C)C(N2CCC(c3ccon3)C2)=O)o1.C12CC1CC(C)C(=O)NC2 C1(N(C(C(CCCC)O)=O)C)CCC2CN(C(c3cccc(Cl)c3F)=O)CC12 C(C)(N=c1[nH]c2c(F)cccc2o1)C1CCN(C(c2c(C)n(C3CC3)cc2)=O)C1 c1(C(N2CCOCC(NC(C34CC(C)(C3)C4)=O)C2)=O)nc2cc(O)ccc2[nH]1 c1(N2CCCC(C(C)NC(c3cc4c(o3)CCCC4)=O)C2)ncnc2scnc12 Cc1cc(C)c(NC(=O)NC(C)Cc2c[nH]c3ccccc23)cc1Br C1(NC(c2snc3ccccc23)=O)CS(=O)(=O)CC1N=c1nc[nH]n2cccc12 C12(NC(CS(CC)(=O)=O)=O)CCCC1N(C(c1cnc(OC)nc1)=O)CC2 C1(CCNC(c2cc(C)sn2)=O)CSCCN1C(=O)CCc1cnn[nH]1 n1(C(C(=O)NC(C)C)C)cc(CC2CCCN2C(=O)C(N2CCNC2=O)C)nn1 Cc1ccc(O)c(C(N2CCC(C(=O)Nc3cccc(C(F)(F)F)c3C)C2)=O)c1 CCC(CC(=O)N(CC(=O)NCCc1ccccn1)C1CC1)C1CCC1 Cc1c[nH]c2ncnc(N3CC4CC(C3)N4C(c3ccc(Br)c(Cl)n3)=O)c12 c1(C(=O)NCCNC(CCC(=O)N(CC)CC)=O)ccc(O)c(N)c1 c1(-c2n(-c3n(C)ccn3)nc(C3CSC3)n2)cc(F)c(Cl)cc1F C1(C(=O)NCC(CNC(C2CC(C)OC2=O)=O)(C)F)CCC=CCCC1 C1(F)(C(=O)NC2C(NC(C3N(C(=O)OC)CCC3)=O)CC2O)CCOCC1 c1(C(N(CC(CC)O)CC)=O)c[nH]nc1CCNC(c1c[nH]c(=N)o1)=O Cc1cccc(CC(=O)NC2C=CCN(C(c3ccn(C)c3)=O)C2)c1Br C12(CNC(C3CCCS3)=O)CCC(CN(C(C3CCCCCCC3)=O)C1)C2 C1(C(C)NC(C2(CCC)CC2)=O)CCCN(C(c2ccc(=O)oc2)=O)C1 N1(C(c2cccc(C3(O)COC3)c2)=O)CC2CCC1C2NC(C1CCOCC1)=O c1(OC)cnc(Cl)c(C(=O)NCC2CCCN(C(c3cc(Cl)ccc3Cl)=O)C2)c1 C1(C(=O)NC(COC)COC)C2CCC(C2)N1C(c1cc2c(s1)CCC2)=O C(=O)(CCCCC(F)(F)F)NC12CC(NC(Cn3c(C)nnn3)=O)C(OC1)C2 Cc1nn(C2CCC2)cc1C(=O)NCC(C(C)C)NC(C1CC12CC2)=O C(CNC(=O)CNC(C1CCSC1)=O)(CC(F)(F)F)NC(C1(COC)CCC1)=O c1(C(N(CC(C)NC(C2=CC(C)(CC)C2)=O)C)=O)cc(F)c2[nH]nnc2c1 n1(CCC(N2CC(C3CN(C(CC(C)OC)=O)C3)C2)=O)cc(C#N)c(O)nc1=O N1(C(CCN2CCN(C)CC2)=O)CCC2CCC(C1)N2C(C1CSC1)=O C1(C)(CNC(=O)C(C)C)CC(OC)CN1C(c1cc(-c2ccccn2)no1)=O N1(C(c2ccc(CC)o2)=O)CC(CNC(C2(CC3CCC3)CC2)=O)C2(CCC2)C1 C1(F)(CNC(c2c(C)ocn2)=O)CCN(C(C2CNC(=O)N2C)=O)CC1 C12(C(=O)NC3CCN(C(C)=O)C3)COC(C1)C(NC(c1ccc(F)cn1)=O)C2 C1(CCNC(c2c(OC)scc2)=O)(NC(=O)CCCN(C)C)CCOCC1 c1(C(=O)NC2C(CNC(C=C(C)C(F)F)=O)COC2)cccc2ccnn12 C1(C(=O)NCC2CCN(C(c3onc(CC)c3C)=O)C2)CCC(=O)N(C)C1 C12(C(N3C(C=C)CCC3)=O)C(NC(c3ccc(C)s3)=O)C3CC1C2C3 C1(NC(C(C)C#N)=O)CN(C(C2CC3(CCOCC3)CO2)=O)CC12CCOCC2 C=C=C(C)CC(=O)NCCCC1CN(C(c2conc2COC)=O)CCO1 c1(OC)ccc(C=CC(N2CCOC(C(=O)N(C)C3CC3)C2)=O)cn1 N1(C(c2onc(C)n2)C)CC2(C)CN(C(=O)CCCC3CCCO3)CC2(C)C1 CN=c1[nH]nc(CC(=O)NC2CC(NC(C3CCC=CCC3)=O)C(O)C2)s1 C1(C(=O)OC(C)(C)C)(C(=O)NC2CC2C(=O)N(C)C)CCCC1.C1(C(=O)N)CC1(F)Cl Clc1cc(N2CCCn3cnnc3C2)c2cc[nH]c2c1 N1(C(CCC(=C)Cl)=O)C2CCCC1CN(C(c1ccn3nccc3n1)=O)C2 C1(NC(C2CCN(C(C)C)CC2)=O)CC(F)CN(C(C2CC=CCO2)=O)C1 C1(C)(C(=O)NCC(CNC(C23OCC(C)(C2)C3)=O)O)CCCNC1=O C12CCN(C1)CC(=O)N2.n1(CC(=O)N(C(C)C(=O)N(C)C)C)cnc(Br)n1 c1(CC)cccc(C(N2CCC(F)C(NC(=O)CSC(C)C)C2)=O)c1O CC(C)(CNC(=O)C(CC1CCC1)n1ccnc1)S(C)(=O)=O c1(C(=O)NCC(C2CCN(C(COC)=O)CC2)C)cc2ccccc2n1C C(=O)(N1CCC(C(N2CCC(C)(N(C)C)CC2)=O)O1)c1nnc(C(C)C)o1 C(=O)(CCC(=O)N1CC(OCCC(=O)NC)C1)NC1(CC#C)CCCC1 NC(=O)C(N)Cn1cccn1.N12CCCC1CNC2=O C1(CC)CCC(C(=O)N(CC(C)NC(c2cnn(CCOC)c2)=O)C)CC1 Cc1nnn(CC(=O)N(CCCCCNC(=O)Cc2cnn(C)c2)C)n1 C1(c2n(CC(CC(C)C)OC(=O)OC(C)(C)C)on2)OCC2CCCC12 N1(C(C(C)SCCCC)=O)CCCC1CNC(c1ccsc1CC(N)=O)=O N1(C(C(C=C)(C)C)=O)CC2CCCC2(CNC(c2ccc(C)o2)=O)C1 C12(CNC(c3c(C(C)C)scn3)=O)CC1CN(C(c1ccc(C(N)=O)cc1)=O)C2 c1(OC)cc(C(=O)Nc2cccc(Br)n2)c(-c2cc(O)ccc2OC)cn1 N1(C(=O)OC(C)(C)C)CC2CC(Nc3cnc(-c4ccccc4F)s3)C1C2 C1(C#N)(C(=O)NCCCCCCN(C)C(c2ccccc2F)=O)CCCOC1 c1(OC)ccc2ncccc2c1C(=O)Nc1cccc(N2CCC2=O)c1 CCCC(C(=O)N1CCCC(N(C(=O)C(O)C2CC2)CC)C1)c1ccc(Cl)cc1 c1(C(=O)NC2CC(C)(NC(=O)CSCc3ccccc3)C2)cc(Br)ccn1 c1(OC(C)=O)cc(NC(c2ccc(F)c(F)c2F)=O)c2ccccc2c1 CCCCC(CC)C(=O)N1CCC(COC)(NC(c2cc(C(C)(C)C)no2)=O)C1 C#CC1(NC(C2(CNC(C3CCOC3CC)=O)CC2)=O)CCC(C)CC1 Cc1nnc(COCC(N2CC(CN(C(=O)CN3CCNC3=O)C)C2)=O)s1 c1(C(=O)NCC2CC(C)N(C(=O)CCCCCF)C2)cc(F)c2ncccc2c1 N1(C(CCOC)=O)CC(C2CCN(C(c3cc(Cl)ccc3C(C)C)=O)CC2)C1 c1(CCC)[nH]ccc1C(=O)NCCCC(C)NC(=O)CC1CC12CC2 N1(C(C(N2C(C)CCC2C)=O)=O)CC2(CC(CN3CCCC3CO)CO2)C1 C=CC(CCC)CC(=O)NC1CN(C(=O)CCCc2ccccn2)CC1O O=C(C1Cc2ccc(Br)cc21)NC12CC(NC(c3nccc(Cl)c3F)=O)(C1)C2 c1(C(=O)NC(CC)(C)CNC(=O)Cn2c(C)c(C)sc2=O)ccc(C)c(C)c1N CC1C(C)N(C(c2cnc3n2CCCC3)=O)CCN1C(c1ccc(Cl)o1)=O c1(C(=O)NC(CC=C)CNC(c2nc(C)oc2OC)=O)cc2c(Cl)cncc2s1 C1(NC(C(=O)NCc2c(C)scc2)=O)CC(=O)N(C2CN(CCN(C)C)C2)C1 C1(C(=O)NCC2CC(F)CN2C(C2CCC(=O)NC2)=O)(COC)CCC(=O)N1 c1(C(N(C(CN(C(C2=C(C)OCC2)=O)C)C)C)=O)cccc2c1OC(C)C2 N1(C(C2=CCC(NC(c3sccc3F)=O)C2)=O)CCc2nc(O)[nH]c2C1 C1(NC(C2(CCCC)CC2)=O)CN(C(=O)CC2(N(C)C)CC2)CC1OC Cc1cnc(CN(C)C(C2(NC(=O)CC3(C)CC3)CC2C)=O)o1 C(=O)(C(O)CCNC(=O)C=Cc1nccs1)N(C)CC1(C)CCCS1 C1(NC(c2cccc(-n3cnnn3)c2)=O)CCCC2CNCC12 C1(O)(CNC(=O)CN)CCCN(C(c2ccsc2)=O)CC1.c1(CC(=O)N)cnoc1 c1(C(=O)NC2CCN(C(c3c(CC)non3)=O)CC2)cccc(OC)c1N c1(CN(C(c2scnc2C)C=O)C(c2cc(C(C)C)no2)=O)ccc(Br)cc1.CO C1(NC(CCC#C)=O)CCCC(NC(=O)C=Cc2nnn(C)n2)C1 CC(C)C(CCN(C(=O)C(C)C1CCC1)C)NC(=O)C(C)(C)O N1(C(=O)Nc2cnc(OC3CCOCC3)cn2)CCC2(CC1)C(F)(F)C21CC1 N1(C(c2cc(C)[nH]c2)=O)CCC(C)C1CNC(c1sccc1-n1ccnn1)=O C1(CC)(CC)CC(C(=O)NCC2CC2C(=O)N(CC(N)=O)CC2CC2)C1 N1(C(C(C=CC)O)=O)CC=C(C(=O)NCc2ccc(C)c(C)n2)C1 N1(C(c2c(C)c[nH]n2)=O)CCC(CC(C)NC(c2cc(Br)n(C)c2)=O)CC1 C1(NC(c2cc(C(F)F)no2)=O)CC2CC(C1)N(C(=O)COc1ccon1)C2 N1(C(C(C)CC2CCCC2)=O)CC2CC1CN2C(c1ccc(C#N)s1)=O c1(NCCN(CC)CC)ccc(S(=O)(=O)N2CCCCC2CO)cc1F C(=O)(CC(C)(C)CCOC)N(C(C(=O)N(CCCC)CCCO)(C)C1CC1)C c1(N2C(CN(C)C(c3ccns3)=O)CCCC2)ccc([N+](=O)[O-])cc1Br c1(C(=O)NCCCC2OCCN(C(CC(C)C(F)F)=O)C2)ccn2cnnc2c1 c1(C(=O)NC2(C3CCN(C(C4C(C)=C4)=O)C3)CC2)nccc2c(C)cccc12 N1(C(C(CC#CC)NC(=O)CC(C)(O)C=C)=O)CCC(O)(C2CC2)CC1 C1(c2onc(C)n2)CN(C(C2CCN(C)CC2)=O)CC(C)O1 n1(CC)cnc(C(=O)NCc2cn(C3CCN(C(C4CC4C(F)F)=O)C3)nn2)n1 c1(C(=O)NCC(C)N(C)C(C2CC(F)(CF)C2)=O)nccnc1C(N)=O C1(SC)CN(C(c2cn(C)nc2C)C(=O)Nc2c(C)cccc2C)CC(=O)N1 CCCC(C)(O)CC(=O)N1CCC(C=CC(=O)NC(C)CCCCO)CC1 c1(-c2cc(C(=O)Nc3ccnc(F)c3)sc2)ccccc1Br N1(C(COCC#C)=O)CCCCCC(NC(c2cc(C(=O)NC)ccc2C)=O)C1 C12(NC(C(c3cn(C)nc3)=O)=O)CC1CN(C(c1ccncc1C1CC1)=O)C2 C=C(C)CC(=O)NCc1cn(C2CCN(C(=O)Cc3cnn(C(C)C)c3)C2)nn1 c1(C(C(=O)OCC)N(C2CCCCC2)C(C(=O)NCC)C)ccc(CC)s1 C1(CNC(c2sc(C)c(-c3ccccc3)n2)=O)CCCN(CC(=O)NCC#N)CC1 c1(CNC(c2ncc(CC)s2)c2nnnn2CCOCC)cccc(O)n1 CC(F)(F)C(C)(C)CC(=O)Nc1ncc(Br)cc1C#N c1(CCS(=O)(=O)NC2C(CC(=O)OCC)CCC2)cc(Br)ccc1F C#Cc1c[nH]nc1C(=O)NCCC(C)NC(=O)Cc1csc(-c2ccsc2)n1 N1(c2nnc(CSC)n2CC2CCCO2)Cc2nnc(C)n2C(c2ccccc2)C1 c1(C(=O)NC(CCN(C(c2c(OC)nn(C)c2)=O)C)C(C)C)cc[nH]c(=N)c1Cl CS(=N)(=O)C1CC(CNC(CCSc2ccco2)C(N)=O)C1 Cc1ccc(C=CC(=O)NCC(CO)NC(c2cc(Cl)cn2C)=O)s1 Cc1cc(=O)n(C)nc1C(N1CC(NC(=O)CN2CCSCC2)CC1CO)=O C(CC(CNC(C1(F)CC=CC1)=O)NC(=O)C(O)CC1CCCCC1)OC CC1=C(c2cc(CN(C)C)cc3[nH]ccc23)CCCC1.C12CCN(CC1)C2 n1(N(C(C2CCN(CC(=O)C(C)=O)CC2)=O)C)nc2c(n1)CCCC2.C1(O)C=CCC1 c1(OC)ccc(CC(=O)NCC(CNC(c2ncc(Cl)cc2F)=O)OC)c(F)c1 C#CCC(CC(=O)NCC1(CCO)CC1)NC(c1csc(C)c1C)=O C12(C(N(C)Cc3c(C)ccs3)=O)CC3CC(C1)CC(O)(C3)C2 C1(C(=O)NCCc2cccc(O)n2)CC2(CC2)CN1C(=O)C(F)n1ccnc1 N1(CC(=O)NC(C)C(C)NC(=O)C2=C(Cl)CC2)CCCCS1(=O)=O C1(NC(N2CC(C=C)C2)=O)CCOC(C(=O)OCC)C1 c1(CC)ccc(C(C)(C)NC(=O)N(CCC2CC3(CC3)C2)C2CC2)cc1 Cc1c(C(N2CCCOC(CNC(C3CCCC(C)C3)=O)C2)=O)nc2sccn12 N1(C(c2c(C(C)(C)C)ocn2)=O)CCN(C(C2CCC2CF)=O)C(CCO)C1 N#Cc1ccc(CNC(C2CCCCN2C(C2CCO2)=O)=O)cc1 c1(C(=O)NC2CC(CCNC(CSc3cn(C)nc3)=O)C2)cc2n(c1)CCOC2 N1(C(C(C)CN(C)C(c2cn(C3CC3)cn2)=O)=O)CCC(C2CC2)C1.N(C)C c1(CC(=O)NCC2CCN(Cc3c[nH]c(Br)c3)CC2)cccc(Cl)n1 N12CCC3(CC1)COC3NC(=O)C2.C12(C(=O)OCC)CC(C(=O)NC)(CCO1)C2 C(=O)(CC(C)(C)C(=O)N1CCCN(C(=O)CC2CCC23CC3)C(C)C1)OC N1(C(C(C2CCC(=O)N2)C)=O)CCN(C(c2ccc(CO)cc2Cl)=O)CC1CO c1(C(=O)NC2CC(NC(C3CCCCC34CC4)=O)C2)cccc2ccnn12 N1(C(c2c(C)onc2Cl)=O)CCC2C(CCCN2C(c2ccnnc2)=O)C1 c1(C(=O)NC(Cc2ccc(C)cc2)(C)CO)cc2ccncc2[nH]1 c1(NC(CC=C)CC(F)F)cc(C)c(S(=O)(=O)N2CCN(C(C)CC)CC2)cn1 c1(-n2c(-c3c(F)ccc(CC)c3)nc(C3CSC3)n2)cc(O)nc2ncccc12 C1(NC(C2C(C)C2)=O)CC2(C1)CN(C(=O)CC1CCC(C(F)(F)F)CC1)C2 c1(C2C(=O)N2)ccc(C(=O)NC(C)(C)C)nc1.C(C(O)CN(C)C(C)C)OCC C(C(F)(C(=O)N1CCC(O)CC1)C(C)C)NC(Cc1cc(C)nn1C)=O CCC(CC(=O)N1CCOC(CNC(c2cnoc2C)=O)C1)CC(C)C C12(C(=O)NC(CCC)C3CC3)CC(CO1)N(C(=O)C=Cc1cc(C)no1)C2 CC(C)(CCC#N)C(=O)N1CCCC(CO)(NC(C2CCCCC(F)(F)C2)=O)C1 c1(CC)ccc(C(C(C)C)NC(=O)CSC2CC2)cc1 C1(NC(c2c(C)sc(O)n2)=O)CCC12CN(C(c1cn3ccnc3s1)=O)C2 C1(NC(C(N2CCSCC2)C)=O)CN(C(=O)CN2CCOC2=O)CC1(C)C C(=O)(C(F)(F)C(F)F)N1CC(NC(c2ccn(CC)n2)=O)(COC)C1 N1(CC)N=C(C(=O)NCCC(C)NC(c2cc3c(nn2)CCC3)=O)CCC1=O n1(CCC(=O)NC2(CNC(c3ccc(C4CC4)cn3)=O)CCC2)cnccc1=O CP(C)(=O)C(O)C(=O)NC1CCC1CNC(c1ccc(NC2CCC2)cc1)=O c1(NC(CCSCC)C)nc(-c2ccsc2)oc1C C12(C(=O)NC(CC(C)(C)C)CO)CC3CC1C2C3(F)F CCC(C(=O)N(CCCNC(c1ncc(F)c(OC)n1)=O)C(C)C)C(C)C C1(CN(C(=O)CSS(C)(=O)=O)C)C2CN(C(=O)CCCC3CCCCC3)CC12 C(c1ccc(C(N2CCN(C)C(C)C2)=O)cc1)=CC(=O)NCCS(CC)(=O)=O c1(OC)ccc(Oc2c(I)cccc2O)cc1C(C)(C)C c1(C(=O)NC2CC(N(C(C=C(COC)C)=O)C)C2)c(Cl)ccc2c[nH]nc12 Cc1nc2ccc(C(N3CCC(C)C3CNC(C3CCC(C)(C)O3)=O)=O)cc2o1 CC1=NC(C)(CNC(=O)CC2C=CC(NC(C3CCCCN3C3CC3)=O)C2)CS1 CC1CN(C(c2ccc(Cl)c(C(F)F)c2)=O)CCCN1C(=O)C#CC1(C)COC1 c1(CC)ncc(C(=O)N(C)CC=CC(=O)NCCC2CCC(C)C2)cn1 C(C(=O)N1CC2C(NC(=O)CN3CCCS3(=O)=O)C2C1)(C(C)C)OCC N1(C(=O)OC(C)(C)C)CCC2(CC1)COCC(CO)O2.C1CC2CCC1C2 C1(=O)C(CCC2CCC2)N1CCO.C1(C(=O)NCC(=O)OCCCC)CC=CCN1 CCC(CC(=O)N1C(C(=O)N(CC(=O)NC(C)C)C)CCC1C(C)C)C1CC1 C(CCCCCN=c1nc(OC)c(F)c(C)[nH]1)N(C(C(C1CC1)OC)=O)C N1(C(C(F)=CCC)=O)CCC(C2CCN(C(c3c(F)cc(F)cc3Cl)=O)C2)C1 CC1C(C)N(C(c2cc(C#N)ccc2O)=O)CCN1C(c1ccoc1)=O Cc1nc2cc(C(=O)NCC3(C(F)F)CCOC3)ccc2s1 C=CCCC(C(=O)NCCC(=O)OCC)N1CCOC(CC)CC1 N1(C(=O)CC2CCCC2)CCC2CC1CN2C(c1cc(O)ccc1Cl)=O N1(C(c2c(OC)cc(Cl)c(Cl)c2)=O)CCC2CN(C(c3c[nH]nc3C)=O)CCC12 C1(NC(=O)Cn2cnnn2)CN(C(C2CC2)=O)C2(CCCC2)C1.n1(C)ccnn1 N1(C(CCCSC)=O)CC=C(CNC(=O)CC2CN3CCC2CC3)CC1 Cc1cnccc1C(C)C(=O)NCC(C)CN(C)C(c1n[nH]cc1Cl)=O c1(CSCC(=O)NC2C(CNC(C=CC(=O)OCC)=O)COC2)ccccc1O CC(CN(C)C)CC(=O)NCC(C)(C)O.C1(N)CC(O)C(O)C1.C1(=O)CN1 N1(C(CCN(C)CC)=O)CCN(C(C2C(C)C2C)=O)CC(C)(C)C1 Cc1ccc(C(C)(F)F)cc1C(=O)NC1(CNC(C2(C)CCCO2)=O)CCOC1 O=C1CN(C(C2CCCN(C(=O)CO)CC2)=O)c2cccc(Cl)c2N1 C1(NC(C2CCN(C)C2)=O)CN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)CCC1CO N1(C(c2ccccn2)=O)CC2CC1CC2N1CC(O)C1 N1(C(CN(C)Cc2ccccc2)=O)CCC(NC(c2c[nH]c(Br)c2)=O)C(F)C1 c1(C(N2CCC(CCNC(=O)CC(F)F)C2)=O)ccnc2[nH]nnc12 c1(C(=O)NC2(C3CCN(C(CCC4C(C)C4)=O)C3)CC2)cc2occc2n1C C1(C(N(C(C)C(=O)O)Cc2cn(CCCC(=O)O)nn2)=O)CCC=CCCC1 c1(SC)ccc(OC(C)C(N2CCC(C)(NC(=O)CSc3nccs3)C2)=O)cc1 c12nc(c(C)s1)C2.N1(C(C=CCCC)=O)CCC(C(C)OCC)C1.OC N1(C(c2c(CC)ncs2)=O)CC(C)CC1CC(=O)NCC12CCN(CC1)C2 C1(C(N(CCCCN(C(c2c(C)cnnc2O)=O)C)C)=O)CCN2CCCC2C1 c1(OCC)cccc(NC(C2(C)CCN2C(=O)C=CC(C)C)=O)c1Cl n1(CC(=O)NCC(CC)(CC)NC(c2ccc(N)cc2C)=O)cc(C)ccc1=O Cc1n[nH]c(C)c1CNC(=O)CC1CCCN1C(=O)C1=NOCC1 C#CC1(C(=O)N(C)C(C2CCCC2)C)CN(C(=O)C=Cc2cncn2C)C1 C12(C(=O)NCc3ccsc3)CCN(C(c3cncc(C4CC4)c3)=O)CCC1C2 c1(OC)cccc(Cl)c1CN=c1[nH]nc(CSC)s1 CC(O)C(C(=O)N(C(=O)NC)Cc1ccnc(Br)c1)NC(=O)C(C)(C)C c1(CNc2c(C)nc(N3CCCC3)cc2)cc(=O)n2ccsc2n1 O(NC(=O)CC(C(C)(C)C)NC(C1(O)CCOC1(C)C)=O)CC1(C)CCC1 n1(CC)nc(C)c(C(=O)NC2CN(C(=O)C(O)CC3CC3)CC2SC)c1C C1(NC(C2COCC(C)O2)=O)CN(C(=O)CC2(C(F)F)CC2)CC12CCCC2 N1(C(COCC=C)=O)CCCC(CC)C1C(N1Cc2c[nH]nc2C1)=O C(c1ccc(Cl)cc1Cl)=CC(N1CC(N(C)Cc2ccc(C#N)cn2)C1)=O c1(C(N2CC3CCN(C(C(CC)(C)C)=O)CC32)=O)cccc2[nH]nc(O)c12 C1(C(=O)OCC)CCN(C(C2(C(=O)NC3(OC)CCOCC3)CC2)=O)CC1CC c1(C(N(C2CCN(C(C3CCC(F)C3)=O)CC2)CC#C)=O)cc2sc(C)cc2[nH]1 C(=O)(C(C)(C)CCCNC(=O)CN1CC(=O)NC1=O)NCC1N(C)CCCC1 C1(C)(C(=O)NC2CN(C(Cn3cc(C(C)=O)nn3)=O)C2)CCCCC1C CCS(=O)CCN=c1[nH][nH]c(=NCCCc2ccccc2C)[nH]1 c1(OC)cc(N)ccc1C(=O)NC1(C)CCN(C(=O)CCCCNC(N)=O)CC1 C(=O)(C1=CCCC1(C)C)NCCC1(C)CCN(C(C(C)C(F)F)=O)C1 C(=O)(CC(CC)C(C)C)N(CCC)CCNC(c1ccnc(SCC(F)F)c1)=O C(=O)(CCCC(F)(F)F)N1CCC(C(C)NC(=O)C(C)(C)CNC(N)=O)C1 Cc1nc(C)n(CC(=O)NCC2CC2CNC(C23CC(C)(C2)C3)=O)n1 S(=O)(=O)(c1ccc(Cl)c(F)c1)N1CCC2(OCCN(C(C3CC(O)CN3)=O)C2)C1 N1(C(C(CSC)C)=O)CCc2cc(CNC(C3CC4C=CC3CC4)=O)ccc2C1 C1(O)(C(C)C)CCCN(C(=O)C(C2CC=CCC2)NC(=O)CCn2cncn2)C1 N1(C(CN2C(C)CCC2C)=O)CCC(CNC(C2CCCCCCC2)=O)C12CC2 C(=O)(C1=NOCC1)NCCC1(CNC(CCc2n(C)ncc2)=O)CC1 c1(OC)cc(CC(=O)NCC(O)CCNC(c2nonc2N)=O)ccc1C=O C(=O)(C#CC1(C)COC1)N1CC(OC)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 C1(C)(C(=O)NC2C(NC(c3scc(C)c3)=O)CCC2)CC(C(F)(F)F)=NO1 N1(C(Cn2nnc(C)n2)=O)CCCC2CN(C(C3CCC(F)CC3)=O)CC12 Cc1cc(C)n(CCC(N2CCC(CC(N3CCOCC3C3CC3CCCO)=O)C2)=O)n1 c1(CC)nc(C)ncc1C(=O)N(CCNC(c1csc(C(F)F)c1)=O)CC N1(C(c2ccc(C(C)(F)F)cc2)C(=O)NC(CC)C)Cc2cnc(CC)nc2C1 N#Cc1cc(CNC(=O)COc2ccc(F)c(Cl)c2)ccc1Br c1(C(N(C(C)CNC(=O)C(O)CCc2ccccc2)C)=O)cccc2ccsc12 C1(OC)CC2(C1)CC(C(N1CCC(CNC(=O)CCSC(F)(F)F)CC1C)=O)C2 Cc1cnc(NCC2CCN(C(=O)CCC3CC3(C)C)C2)nc1 c1(N2CC3CC(NC(c4n(C)ncn4)=O)C3C2)ncc2c(n1)CCOC2 C1(CNC(C2CCC(=O)O2)=O)CC(F)CN1C(=O)CC1CCC(C(F)(F)F)O1 c1(-c2ccc(-c3ccc(C(N(CC(=O)O)C)=O)cc3)o2)cccc(C#N)c1 N#CC1(C(=O)NC2CC(NC(=O)Cc3nocc3C(C)C)C2)CCCOC1 CC1CCN(C(=O)C(C)(C)C(N)=O)CC1NC(=O)Cc1cc(F)ccc1F C12(C(=O)NCC3N(C)CCN(C(c4nn[nH]c4Cl)=O)C3)C3CCC(CC13)C2(F)F c1(C(=O)NCCC(C)CCNC(=O)CCN2CCC(F)C2)cccc2[nH]ncc12 C12(CC(=O)NCCn3cc(CNC(c4cc(O)no4)=O)nn3)CCC(CC1)C2 c1(CCCNC(C(C)(C)OCC)c2ccccc2)ccc(NC)cc1 c1(C(=O)NC2CC(C)(CNC(C3N(C)CCOC3)=O)C2)cccc2cn[nH]c12 c1(C(=O)NC(C2CCN(C(c3cc(C)oc3)=O)CC2)C)ccc2[nH]ccc2c1 c1(C(=O)NCCOC(CNC(CCOCC)=O)(C)C)cncc2c[nH]nc12 N1(C(COC)=O)CCC2(CC1)OCCc1cc(C(=O)NCC(C)C)sc12 C1(NCC(C2CC2)NC(=O)OCC)CC1(Br)Br C(=O)(CCCN=[N+]=[N-])NC1CCC(C(=O)NCc2c(COC)noc2)CC1 c1(C(N2C(C)(CNC(CC3(C(=C)F)CCC3)=O)CCC2)=O)cnc2ccoc2c1 C(N=c1cc[nH]cc1C#N)C1C(C(F)(F)F)CCN(C(C(C)CC(C)(C)C)=O)C1 C=C(Cl)CC(C(=O)N1C2CCC1CC2)NC(C1CCNC1=O)=O C=CC1(C(=O)NC2CCC(C)(C)C(C)C2)CCN(C(C2OCCC2C)=O)CC1 C1(NC(CC2(C(=O)OC)CC2)=O)COC2(C1)CN(C(c1ccc(C)nn1)=O)C2 C#CC1CN(C(c2coc(Cl)n2)=O)CCN1C(c1csc(O)n1)=O c1(C(N2C(C(C)NC(C(C)OC)=O)CCC2)=O)cc(Br)c(C)s1 C1(NC(=O)CNS(=O)(=O)C2CC2)CN(C(C2CC2(F)F)=O)CC1C(F)(F)F N1(C(C(C)(C)CCl)=O)CC(C(=O)NCc2ccco2)CC(F)(F)C1 CC(C)C(C#N)C(=O)NC1(CCCCNC(=O)NC2Cc3nccn3C2)CC1 CC1C(=O)NC(=O)CN1C(=O)CC(C(F)(F)F)NC(=O)CCc1nncn1C CC(C)CCC(=O)C(=O)N1CC(n2cc(-c3cccc(OC(C)C)c3)nn2)C1 c1(C(N2C(c3scc(CC)n3)CCC2)=O)c[nH]c2c(-c3nn[nH]n3)cccc12 c1(C(=O)NC2(CC=C)CCN(C(c3coc(C)n3)=O)C2)sc2ccccc2c1C O=C(C=C(Cl)Cl)NCC(O)CCNC(=O)Cn1cc(C2CC2)cn1 Cc1ccc(C(=O)NCC2CC(F)(CNC(=O)COC(F)F)C2)c(F)c1 CC1Sc2ccccc2N(S(=O)(=O)c2cnnn2C)C1C c1(C(=O)NCCC2CCC(NC(c3c(C)noc3)=O)C2)cncc(F)c1Cl C1(NC(C(CCSC)OC)=O)CCC2CCCC1O2.C12(CCC1)C(=O)N2 CCCCC(F)C(=O)N(C)CCN(C(=O)CC(CC1CCCC1)CC)C c1(C(N2CCC(NC(C(CSC)C)=O)C2)=O)cnc2[nH]c(C3CC3)cc2c1 C(=O)(CCP(C)(C)=O)NCC(CCOC)NC(C1CS(=O)(=O)CCO1)=O c1(C(=O)NC2CCC(NC(C3ON=C(C)C3)=O)C2)c[nH]c2cccc([N+](=O)[O-])c12 N1(C(c2cc(C)no2)=O)CCOCC(CNC(=O)CN(c2cnccn2)C)C1 c1(OC)cccc(OC)c1C(N1CCC(C)(C(=O)NCC2(O)COC2)CC1)=O C1(CNC(CCNC(=O)CO)=O)CCCN(C(c2ccccc2C2CCC2)=O)C1 c1(C(N(C2CCC(NC(=O)CCCC#N)CC2)C)=O)cccc2ccn(C)c12 n1(CCC)c(C)cc(C(=O)NCC2CC2NC(C2(N3CCCC3)CCC2)=O)c1C C1(NCc2ccc(OC)nc2)CC2(C1)CC(CC(=O)CSc1nnnn1C)C2 c1(C(N(C)CC2CCCN2C(c2cnn(C)c2)=O)=O)cc(N)cc(O)c1 N1(C(CC2C(C)(C)OCC2)=O)CCN(C(c2cnc(Cl)s2)=O)C(C(C)(C)C)C1 N1(C(CCC(=O)NC)=O)CCCCC(CCC(N2CCC(C#N)C2)=O)C1 Cc1ccncc1-c1cn(CC(F)(F)CNC(C2CC(OC3CC3)C2)=O)nn1 C(=O)(C1CCCc2ccnn21)NC1CC(NC(C=Cc2n(CC)ccn2)=O)C1 C1(N(C)C(C2CCC(=O)N2)=O)CCCN(C(C23CC(C)(CO2)C3)=O)C1 C(CCCS(=O)(=O)NCc1cccc(OC)c1OC)OC CCS(=O)(=O)CC(=O)N1CCC(c2n[nH]c(CNC(=O)CC(C)(C)O)n2)CC1 Cc1nn(C)c(-n2cncn2)c1C(=O)OC1CCCCC1C O(NC(=O)CCCCCn1cc(C(O)C2CC2)nn1)C(C1CC2CCC1CC2)=O C1(CNC(c2ccc(CC)[nH]2)=O)CC(N(C)C)C1(C)C.c12cc(ncn1)C(=O)N2 N1(C(CCC(C)SC)=O)CCC2(CCC(NC(=O)C(CC)N(C)C)C2)C1 Cc1ccc(Cl)cc1OCCC(=O)Nc1nccc(Cl)c1C C1(C(CO)CC)CCCCCC1.n1(CC(=O)NNS(N)(=O)=O)cc(CCCSC)nn1 c1(C(N2C3CC(NC(CC(C)OC)=O)C3CC2)=O)cc2c(C(F)F)nn(C)c2s1 c12ccc(O)c(c1)CCNCC1CCN(C1)C(=O)N2.CN1CCN(CCN)CC1 c1(C(=O)NCC2C(NC(C(CCOC)C)=O)CCC2)ccc(C)c(OC)c1F N(C(=NCCF)N1CCC(c2ccccc2F)C1)CC1CCC(=O)NC1 C#CC1CCCN(c2nnc(C3CCC(=O)N3)n2CC2CC3(CC3)S(=O)(=O)N2)C1 CCC(CNC(c1ccccc1OC1CC1)=O)N=c1[nH]nc(CCOC)s1 CC(C)(C)C1=CCN(C(=O)CC(C(C)(C)C)NC(C2CCC3(CCC3)O2)=O)CC1 C1(C(=O)NCCN(C(c2scc(COC)c2)=O)C)CC1C1CCC1 C1(C(N(C)CCC2CC2)=O)CCCN(C(C2Cc3nccn3C2)=O)CC1 C(=O)(C(CC)C(C)(C)CC)NC1CCCC(NC(c2onc(CC)c2C)=O)C1 c1(C(=O)NCC2CCC(C)N(C(=O)COC(F)F)C2)cccc2nc(O)ccc12 CC1CCCCN(C(C23CC2CN(C(=O)C(c2cccc(Cl)c2)N(C)C)C3)=O)C1 C1(CCN(C(=O)NC(COCC)C)CCOC)CCCC(C)C1 n1(C(C(=O)N(CCNC(=O)CCN2CCC2)CC)C)cnc(C#N)n1 c1(C(=O)NC2C(C)CCN(C(c3cnc[nH]3)=O)C2)cc2ccccc2c(=O)o1 C(=O)(C(C)CC(F)(F)F)NC(CCN(C(c1ccc(SCCC)cc1)=O)C)C C1(n2cc(CC(C(=O)OC)NC(C3CC(O)C3)=O)nn2)CCCC(C)C1 N1(CCNC(C2(C(=O)OC)CC2C)=O)CCOC(C(=O)N)C1.C(CO)CC C1(CC=C)(CNC(C2CC=CC2)=O)CCN(C(=O)CS)C1.C1(CO)(CO)CC1(C)C C1(NC(c2c(C)occ2)=O)CCCN(c2ccnc(C3CCC3)n2)C1 N1(C(CCOC(C)=O)=O)CC(NC(c2cn(C)nc2SC(C)C)=O)C2(CCC2)C1 C#Cc1cc(C(N2CCOC(C)(CNC(=O)CN3CCC3C)C2)=O)cc(F)c1 N1(C(C(CC#C)C2CC2)=O)CCC2(C=C(C(=O)Nc3ccccc3C)C2)C1 c1(NCCOCCN(C)C(C2CC3CC2C2CC32)=O)cnc(C#N)c(C#N)n1 C(CC(C(=O)Nc1cscc1C)NC(C1CC(C)(C)C1)=O)OCC C1(CNC(C2C(CC)CCC2)=O)CN(C(C2CCC(N(C)C)C2)=O)CCC1(C)C c1(NCCOCC(=C)C)[nH]c(=NC2CCN(CC)CC2C)nc2ccc(OC)cc12 c1(-c2c(OC)cc(CN3CC4(COC4)C3)cc2)ccc(C2=CCC(O)CC2)cc1 N1(C(CNC(=O)CNC(=O)CC2CCCC3CC23)=O)CC2C(C1)C2(F)F CC(C)(CC#N)C(=O)N1CCN(CCNC(C2CCCN2C2CCCC2)=O)CC1 O=S(=O)(C1CCCC1)NC1CCN(CC2CCCCC2)C1 CCC(C(=O)NCCN(C(c1cn(C)c2ccccc12)=O)C(C)C)C(C)(F)F CCCC(C(=O)NC1COCC1NC(=O)C=Cc1sccc1C)NC(C)=O O=C(C(CCc1ccccn1)N1CCCCC1c1ccc(O)cc1)NCCCF C1(NC(C(C)(C)OCC)=O)CC(C2CCN(C(=O)Cc3ccnn3C(C)C)C2)C1 N1(C(CC(CC)C)=O)CCOC2CN(C(c3cccc(C4CC4)c3)=O)CC12 C1(NC(C2(OC3(OC)CC3)CCCC2)=O)CN(C(=O)CCOCC(C)C)CCO1 CC1OCCN(C(=O)CCn2ccnc2)C1C(=O)NCCC[Si](C)(C)C C1(NC(CCC(C)CN(C)C)=O)CN(C(=O)CCCCCF)CC1C1CC1 c1(C2(NC(C)C(=O)Nc3cncc(Br)c3)CC2)cccc(C#N)n1 C1(CNC(C=C(C)C)=O)CN(C(=O)Cc2cccc(C)c2)CC(C)(C)C1 c1(C(CNC(=O)CC2(O)CCC2)NC(C2C(CC)CCO2)=O)ccc(F)cc1F N1(C(CNS(CCCC)(=O)=O)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C(CO)C1 Cc1cnc(NC(C2CC3CC3N2C(C2CNC(=O)O2)=O)=O)c(C)n1 C1(C)(C(=O)NCC(C)N(C)C(c2ccc(-n3ccnc3)cc2)=O)CCCOC1 N1(C(CNC(=O)C=CCn2cncn2)=O)CC2CCC(C1)C(=O)O2 CC1(CCO)CCN(C(C2CCCCC2NC(c2cccc(CC#N)c2)=O)=O)C1 N1(C(C(C2CCCO2)NC(=O)Cn2nccn2)=O)CCCC2(CC1)CC2 N(C1CCCc2ccccc21)C1CN(c2nccc(N3Cc4n(C)cnc4CC3)n2)C1 C(=O)(C1=CC2(CCOC2)C1)NCCCCCC(=O)N1CCC(C(N(C)C)=O)C1 c1(O)ccc2c(c1)OCO2.CCCC(CC(=O)OCC)OC C1(N(C(COC)=O)C)CN(C(=O)C(c2cccc(Cl)c2)C)CC1O C1(C(C)(C)NC(C2C(C)C2)=O)CCN(C(=O)CC(C)(C)F)CC1 C1(O)(CNC(CCC)=O)CC(CNC(C2CCOC2CC)=O)C1 c1(C(N(CCNC(=O)C=CC2CC2)CC)=O)cc2c(cc1N)OCCO2 Nc1cc(C(=O)NCCCNC(=O)CNC(=O)CC(F)(F)F)c(F)c(O)c1 C1(C2(O)CN(C(=O)C(O)Cn3cncn3)C2)(CNC(C2C(=O)OCC2)=O)CC1 C1(NC(C(C)N(C)C)=O)CN(C(c2ccc(Cl)cc2)=O)CC12CCCC2 CC1(C(=O)N(CC(=O)NCC(F)F)CC2(CF)CC2)CCCC1 O=C(C1=CC2(CCOC2)C1)N1CC2CC(C1)N2C(c1ccc2ncccc2c1)=O N1(C(C2(N(C)C)CCCSC2)=O)CC2(C)CC1(C(N1CC3(C1)CN(C1CC1)C3)=O)C2 C(C)(N=c1[nH]c(=NCCC(C)c2cn[nH]c2)[nH]c2ccsc12)c1ncc(C)cc1Br c12nc(-c3ccsc3)nn1C2.n1(C(F)F)ccc(C2CC2)n1 C1(CC)(NC(C2C3COCC23)=O)CCCN(C(C2CC(=C3CC3)C2)=O)C1 C1(CC#C)(NC(C2(C)C=CCN2C(C2COC(C)C2)=O)=O)CCCCC1 C1(CNC(CC(C)(C)SC)=O)CN(C)CCN1C(C1CC2(C1)CC(CO)C2)=O C#CCCCC(=O)NCC(C(=O)NCCCc1c[nH]nc1C)N(C)C Cc1ccnc(C)c1C(=O)NCCN(C(=O)C1=CCOC1)C(C)C C1(NC(c2ncc(C)c(Cl)c2)=O)C(C)CCN(C(=O)COCc2ccncc2)C1C C1(C)(NC(C(C2COC(C)(C)O2)O)=O)CCCN(C(=O)C=CCn2cncn2)C1 c1(C(N2CCC(CN(C)C(c3cc(N)ccn3)=O)CC2)=O)c(F)ccc(Cl)c1F C=CC(C)(CC)C(=O)OCC(=O)Nc1csc(-c2ccc(Cl)cc2)n1 C(N=c1[nH]c(=NC2CCSC2)[nH]c2c1COCC2)C1CC(OC(C)(C)C)C1 c1(C(N2CCC3CN(C(CCC(C)OC)=O)CC32)=O)ccc2nc(C)[nH]c2c1 S(=O)(=O)(c1c[nH]ccc1=NC1CCC2(CCC2)C1)NCC1(C)CCCCO1 CC1CCC(CNC(=O)Cn2ncccc2=O)N(C(c2csc(S)n2)=O)C1 C(C(O)(C(=O)N1CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1)C(F)(F)F)N(C)C CC(C)CC(C)C(=O)NC1(C)CCN(C(C2CCCC3(CC3)C2)=O)C1 c1(C(c2nnnn2CCCF)NCCCNC(N)=O)sncc1Br.c1(N)ccccc1 C1(SCC)CCC(c2nnnn2CCCC2CC2)(NCCC(C)(C)C(C)C)CC1 c1(C(=O)NCC2(C)CCC(NC(=O)C(O)C(F)F)CC2)nccc2ccccc12 C1(C(=O)NCCCN(CCCNC(c2ccc(C#N)[nH]2)=O)C)CCCNS1(=O)=O CC1(C)CC2(CC2C(=O)NCC2C3CN(C(=O)C=Cc4ccc[nH]4)CC23)C1 c1(C(=O)NCC2CC(NC(=O)CCSc3ccccn3)C2)cc2c(s1)CCC2 N1(SCC)CCCC(C2CN(c3cc(N4CCCC(CO)C4)ncn3)C2)C1 C1(NCc2c(C)cccn2)CC2(C1)CC(NC(C1CCNC(=O)C1)=O)C2 N1(C(CSCC(N)=O)=O)CCOCC12COCCN(C(c1cnoc1)=O)C2 n1(CC)nc(CNC(C2(NC(=O)CCCC3CCC3)CCCC2C)=O)c(C)n1 C#Cc1ccnc(C(N2CC(O)(C3CCCN3C(C3COC(C)(C)C3)=O)C2)=O)c1 C1(C(N(CC(=O)NCC2CCC(NC(=O)C3CC3)C2)C)=O)CCCCC12CCC2 C=C(Cl)CCC(=O)NCC1CN(C(=O)Cc2coc(C(F)F)n2)CC1O CC1C(NC(C2(CCF)COC2)=O)CCN1C(c1ccc(OC(F)(F)F)cc1)=O C(CC(=O)N(c1ccsc1)C)(C(C)C)NC(C(=O)NCC)=O N1(C(CS(=O)(=O)NC(C)(C)C)=O)CCCC(O)(CCNC(=O)C(O)C(C)(C)C)C1 C=CC(CC)CC(=O)NC(C)CCC(=O)NCC1CCC1C(=O)OC C(=O)(CCC(C)(C)C)N(CC(CC)NC(c1cccc(C)n1)=O)C CN1CCN(CCC(=O)NC2CCN(C(=O)CC3(O)CCCOC3)C2)CC1 C1(CC)CN(C(c2cc(C(C)=O)n(C)c2)=O)CCN1C(=O)C(=O)NC(C)C C(C)(C)(CCC(=O)NCCCCCC(=O)Nc1cnccc1C)OC c1(OC)ccc(C(=O)N(CC(C)NC(c2csc(C3CC3)n2)=O)C)c(Cl)n1 N1(C(=O)CC(O)C2CCCC2)CCC2(CC1)CN(C(=O)C(F)(F)C1CCCC1)C2 c1(C(N(C2CCN(C(=O)C(C3CCCC3)OC)C2)CC#C)=O)nccnc1OC c1(C(=O)NCC(C)NC(=O)CC(C)n2cccc2)cccc(N2CCOC2=O)c1 c1(OCCC#C)ccc(C(=O)NCC2CCC(NC(=O)C(COC)OC)C2)cc1 C1(C(=O)NCc2cnn(-c3cccc(Br)c3)c2)CCCC2(CNC2)O1 N1(C(CC2C(OCC)COCC2)=O)CCC(C)C(CNC(=O)C(C)C#N)C1 C12(C(=O)NC3C(OC)CN(C(CC4C(OC)CC4)=O)C3)CNCC1COC2 c1(C(=O)NCCN(CCC)Cc2ncc(C)o2)cc(C)oc1C CC1CN(C(=O)C2=CCCS2)CC2(CCN(C(=O)CCS(C)=O)C2)O1 c1(C(N2CCN(C(c3c(C)ncs3)=O)C(C3CC3)C2)=O)noc2ccc(F)cc12 N1(C(C(C)C(C)O)=O)CC2CCC1C1CN(C(c3cc(Cl)n(C)n3)=O)CC21 Cc1ccc(N)c(C(=O)NC2(CNC(c3n[nH]cc3C3CCC3)=O)CC2)c1 c1(C2(C(N)=O)CCC2)ccc(NC(=O)Cc2ccc(Cl)cc2)c(F)c1 N1(C(c2ccn(CC)n2)=O)CCCC(C2CCN(c3nccnc3F)CC2)C1.C1CC1 c1(C(N2CC3CC(NC(Cn4cnc(OC)n4)=O)C3C2)=O)cnc2ncccn12 C1(C(=O)NC2(CN(C)C)CC2)CN(C(=O)C(F)C2CC2)CC12CC2 N1(c2nc(=N)[nH]c(=NCc3ccccc3CC(N)=O)[nH]2)CCC2(CCC(O)C2)C1 C(=O)(C(F)(F)C1=CCOCC1)NC1C=CCN(C(c2cncc([N+](=O)[O-])c2)=O)C1 CCC(C)CC(=O)C(=O)NC12CC(C(N3CCSC(C)(C)C3)=O)(C1)C2 C1(NC(c2nc(C)ccc2Br)c2n(CCCC)nnn2)CS(=O)(=O)C12CCCC2 N1(CC(=O)N(C)C)CCN(C(C2CC2F)=O)C1=O Cn1c(C(N2CC(F)(CNC(C3CCNC(=O)C3)=O)C2)=O)cc2ccccc12 Cc1cc(C2CN(C(=O)NC(c3cc(C4CC4)no3)C)C2)no1 c1(C(C)=O)ncc(Br)cc1NC(=O)CC1CCCN1Cc1cc(C)nn1C N1(C(=O)CCc2cncs2)CCC2C(C1)CN2C(=O)CCCc1ccccn1 C(=O)(C1Cc2ccc(Cl)cc21)NC(C1CN(C(c2c(C)ccc(OC)c2)=O)C1)C N1(C(CC=CCC)=O)CCCCC1C(=O)NC(CC1CC1)CO Cc1csc(C(=O)N(C2CC(NC(c3ncn(C)c3C)=O)C2)C)c1Br c1(C(C(=O)NCc2cncc(Br)c2)N(CC(=O)NCC)C)cnc(OC)cc1C C1(NC(C(=O)N(C)Cc2cc(Br)ccc2F)=O)CC2(CCCCN2)C1 C(=O)(CCCS(C)(=O)=O)N1C(C)C(NC(C2CC(N(C)C)C2)=O)CCC1 c1(C(=O)NCC2N(C(CSc3nc(C)[nH]n3)=O)CC=C2)cc(F)ccc1Br CCC(C)C(C(=O)N1CCC(Sc2nn[nH]n2)CC1)c1ccccc1 C1(NC(c2c(C)nccn2)=O)(CO)CCCN(C(=O)C(c2ccn(C)c2)C)C1 C1(CNC(C(C)=C(CC)C)=O)CC2(CCC2)CN1C(=O)C(CC)C(C)C N1(C(c2c(CSCC)cccc2)=O)CC2CN(C(c3[nH]c(C)nc3C)=O)CC2C1 c1(OC)ncc(C(=O)Nc2cnn(C3OCOC3)c2)cc1-c1cncc(C#N)c1 c1(CC)nn(C)c(Cl)c1C(=O)NCC(C1CC1)NC(=O)CCc1ccnc(C)n1 S(=O)(=O)(c1c[nH]c(C(=O)NC2CC(NC(C3CCC4C3C4(F)F)=O)C2)c1)N(C)C c1(C(=O)NC2CC(NC(c3c(C)n[nH]c3C)=O)C2)cc2n(n1)CC(C)NC2 c1(C(=O)NC(CCC)C)ccc(C)c(O)c1O c1(C(c2n(CC(=C)C)nnn2)NCc2nc(Br)cs2)ccc(Br)c(C)c1 Cc1ccc(C(N2CCC3CN(C(C4CC(=O)NC4(C)C)=O)C3C2)=O)c(F)c1F n1(CCC(=O)N(CCNC(CCCOC(C)C)=O)C2CC2)ccc(O)nc1=O c1(C(=O)OC)nccnc1C(=O)NC1COCC1NC(c1cnc(S)nc1)=O N1(C(CCc2scc(C)n2)=O)CC2CC(NC(C3NC(=O)CC3C)=O)CC1C2 C1(NC(C2N(S(C)(=O)=O)CCC2)=O)CC(F)CN(C(C2C3CC4C(C3=O)C24)=O)C1 c1(NC(C2(C)N(C(c3n(C)cnn3)=O)CC2)=O)cncnc1Br C1(C(N2CC(C3(NC(C4CC45CC5)=O)CC3)C2)=O)CCc2ccnn2C1 Cc1cnc(N2CCN(C(c3cc(I)cc(F)c3F)=O)CC2)c([N+](=O)[O-])c1 CC1CCN2C1C(=O)N1C(CCC1)C2=O.c1(CNC(N)=O)cccc(CO)n1 N1(C(C2CCC(N(C)C)C2)=O)CC2(CNC(=O)CCCC3CCC3)CC1CO2 c1(NC(C(=O)NC(Cc2c(C)nc(SCC)s2)=O)=O)c(F)cccc1F C(C)(CCC(=O)NCCC1COCCN1C(=O)CCOC(=O)NC)OC.OC [N-]=[N+]=NCCCCCC(=O)N1CC2(CNC(c3cc(C(F)F)[nH]n3)=O)CC1CO2 c12c(cccc1C)CN=C(NCCc1cccs1)NCCN2C.n1(CC)cnnn1 c1(C(=O)NC23CN(C(C4C(OCC)C4)=O)C(C2)C3)cn(C)c2ccccc2c1=O CN1CCCC(C(=O)NCC2(NC(=O)CCc3cn(C)cn3)CCC2)C1 c1(C(=O)NCC2(F)CC(CNC(CN(CC(C)(C)C)C)=O)C2)cccc(F)c1F CN1CC(=O)N(CC(=O)NCCC2CN(C(c3cc(F)cs3)=O)CCO2)C1=O c1(CC)onc(OCC(=O)NCC2(O)CCN(C(=O)Cc3ccnn3C)C2)c1C C12(CNC(c3c(C)nc[nH]3)=O)CCCC1CCN2C(C1CCc2nn[nH]c2C1)=O c1(C(N2CCN(C(C(CCC)=CC)=O)C(C)C2)=O)ccc2c(C)[nH]nc2c1 c1(OCC)oc(C)nc1C(=O)NCCNC(c1cccnc1S)=O N1(C(C(C)SCC)=O)CC2C(CNC(c3ccccc3CC)=O)C2C1 C1(C)(C(=O)NC(CC)CNC(c2cnn(C)c2Br)=O)CCCC1(F)F c1(C(N(C(C)C(=O)N(C(C)CC(F)(F)F)C)CC)=O)cccc(O)c1F C1(C(=O)SC2C(C(N(C3CCN(C4CC4)C3)C)=O)CCC2)CCOC1(C)C c1(OC)ccc(C(=O)NCCC2CCN(C(c3cnccc3N(C)C)=O)C2)cc1 c1(C(N2C(C(=O)Nc3ncn(C)c3)CC3(CC3)C2)=O)ccc2c(c1)ncn2C c1(CC(=O)NC2C(NC(COCCC=C)=O)CC2)ccc(C(C)(C)C)cc1 C1(NC(c2c(C)nc(CC(C)C)o2)=O)CC2CC1N(C(c1ncc[nH]c1=O)=O)C2 N1(C(C2(CC(=O)OC)CC2)=O)CC2CC(NC(=O)CNS(=O)(=O)NC)C1C2 C1(C(=O)NCC(CNC(Cn2c(C(C)C)ncc2)=O)CO)CCCCCC1 C1(NC(C(CC)CC2CCCC2)=O)CC2(CCN(C(=O)Cc3ccsc3)C2)C1 C1(CC=C)(C(=O)NCCC(=O)N(C)CC)CCN(C(=O)CC2CCCC2)C1 c1(C(N2CCC(C)(NC(CCCCC#C)=O)C2)=O)cccc2occ(Br)c12 C1(NC(CC=C)=O)CC(N=c2[nH]c3c(C)cccc3o2)C12CCOCC2 c1(C(=O)NC(CNC(c2[nH]cc(C(C)=O)c2)=O)(C)C)cnc(C(F)F)nc1 C1(C(N2CC(CNC(c3cc(C4CC4)n(CC)n3)=O)C2)=O)CCC2CCC(=O)N12 c1(C(N2C(C3CCN(C(=O)NC)C3)CCCC2)=O)ccc2c(c1)CCC(C)N2 c1(C(=O)OCC)cc(CNCC(C)CC(N2CC(N(C)C)C(O)C2)=O)oc1C CC1CCCN(C(=O)CCc2cnc[nH]2)C1CNC(C1CCCS1)=O CS(=O)(=O)CCC(=O)NC12CC1CN(C(c1cc3occc3s1)=O)C2 N1(C(c2c(C)n(C)c(C(C)(C)C)c2)=O)CC2=C(C1)CN(C(C13CCC1C3)=O)C2 c1(C(N(C)CC2(O)CN(C(CC3CC(CC)OCC3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 CN1CCC2CN(C(c3ccc(-c4cnn(C)c4)s3)C(=O)NCCSC)CCC12 C1(C(=O)NC(CC)C(=O)NC)(C(C)C)CCN(C(c2nnccc2C)=O)C1 C1(NC(C2(CCC=C)CN(C(=O)CCCC=C)C2)=O)CCCCC1C(=O)NC C1(C(=O)NCC2C(C)CC2)CCC(NC(C2CCCS2)=O)C1 c1(C(C(N2CC(C)(CN3CCCC3)C(O)C2)=O)(C)C)ccc(C#N)c(F)c1 C1(NC(C(C)OCCOCC)=O)CC2C(NC(=O)C(C)(C)Cl)C2C1 Cc1cccc(C)c1C(O)C(=O)NC1COCCC1NC(c1cnc(Cl)[nH]1)=O C1(COC)CN(C(c2cc(CNC(=O)C(C)C#N)[nH]n2)=O)C1(C)C CC1(C2(C(=O)NC3C=CC(C(=O)NC(c4ccco4)CO)C3)CC2)CC1 C1(C(=O)NCC2(F)CC(CNC(C3CC4CCC3C4)=O)C2)CCCC12CC2 c1(CC)n[nH]c(CC)c1CC(=O)NC(CNC(C1COCCO1)=O)C(C)C O=C1CC2C(CCCN2C(C2(CF)CCN(C(c3ccc([N+](=O)[O-])o3)=O)C2)=O)N1 N1(C(CNC(=O)OCC)=O)CCCN(C(c2c(F)cccc2Br)=O)C(C)C1 c1(OC)ccccc1-n1ccc(C(N2CCOCC2CNC(C2CC2F)=O)=O)n1 C(=O)(CCCS(N)(=O)=O)NC1C(CNC(CC2ON=C(C)C2)=O)CC1 C1(NC(Cc2c(N)nccc2)=O)CN(C(c2cnncc2O)=O)C2(CCCC2)C1 CC(O)C(C)C(=O)NCC1(CNC(c2ncnn2C2CCOCC2)=O)CCC1 O=S(=O)(c1cccc(=NC2CCOC2)[nH]1)N1CCC=C(Cl)C1 C(=O)(C#CC1CCCO1)NC1(CC=C)CCN(C(=O)C=CCC2CCCC2)C1 N1(C(c2ccc(C(=O)OC)cc2)=O)CC2CN(C(C3CC(O)C3)=O)CC2C1 Cc1ccc(NCc2ccc(Oc3ccc(C#N)cc3)cc2)c(Br)c1F c1(C(=O)NC(C(C(C)C)C)CNC(=O)C=CCO)cc2ccccc2c(O)n1 C(=O)(C(F)(F)C(C)O)N1CC(C(NOCC(=O)OCC)=O)C(C)C1 c1(SCC(=O)NCCOC2CN(C(C=C(CC)C)=O)C2)nnc(C)n1C c1(N)ccc(O)cn1.C1(C(=O)NCC2CCCC2C)(COC)CC(=O)C1 C12(CNC(CNC(=O)NC)=O)CCC(CC1)N(C(C1(C)CCCC1C(N)=O)=O)C2 C(=O)(C(CCNC(=O)Cc1csc(C)n1)CC1CC1)NCC(C1CCCC1)OC C1(C(N2C(CCNC(C3CN4CCC3CC4)=O)CCC2)=O)CCCCC1C1CC1 C1(NC(CC2CC(=C)C2)=O)CN(C(c2c(C)cccc2Br)=O)CC12CCC2 C1(C(=O)NCC2(C)CCN(C)CC2)CCN(C(=O)CCS(C)(=O)=O)C12CCC2 C1(NC(C2C(CC)CCC2)=O)CCN(C(=O)Cc2sc(C)nc2C)CCC1(F)F c1(C(=O)NC2C=CC(C(=O)NCC(C(=O)OC)C)C2)cnn2ccccc12 Cc1cccc(C)c1CNC(=O)CC(C(C)C)NC(C1(C)CC1(C)C)=O N1(C(C=CCC)=O)CCCC12CCN(C(c1cc(CC)cc(Cl)c1)=O)C2 c1(COCCN2CCC(=O)N(CCCCCCCC)C2=O)ccc(Cl)c(Br)c1F N1(CCC)CC2CCC(C1)CC2NC(c1cccc(OC)n1)=O c1(OC)ccc(CN(C2CC3(CCNCC3)C2)C(=O)C(C)(O)CCl)c(C)c1C CS(=O)CCC(=O)NC1CN(C(c2cc(N3CCOCC3)ncn2)=O)C1 CC1(C(=O)Nc2nc(C(N3CCCN(CCO)CC3)=O)co2)CCC2CC2C1 CC(C)C(C)CC(=O)NC1CCN(C(C2CC=CC(O)C2)=O)CC1CO Cc1nn(CC(N2CC(C(C)NC(c3nc(Cl)oc3C)=O)C2)=O)c(C)c1Br c1(NC(C(CC)NC(C2CC(N3CCN(C)CC3)C2)=O)=O)ccc(F)cc1 Cn1cnc2c(NC3CCC(O)(c4ccccc4)CC3)nc(S(C)(=O)=O)nc12 c1(C(=O)NCC(CCNC(c2cc(CCC)n(C)n2)=O)O)ccc(F)c(CC)c1 C1(N2CC2=O)CC12CCC2.C1(C)CCCCC1.C1(CC#N)CCCC1 CCC(CC)CCC(=O)NCC1(NC(=O)C(n2cc(C)cn2)C)CC(OC)C1 c1(C(C(=O)NC2CC(NC(C3(CC=C)CC=CC3)=O)C2)(C)C)ccc(CC)cc1 C1(=CC(=O)NCCC2CCC(NC3COCCO3)C2)C2CC3CC(C2)CC1C3 CC1CCC(CC(N2CCC2CNC(=O)CC2(N3CCOCC3)CCCC2)=O)C1 c1(C(C(=O)NC2C(C)CN(C(=O)Cc3cnc[nH]3)C2)=O)ccc(F)c(F)c1 N1(C(Cc2ccc(C)s2)=O)CCC2(CC1)CC(NC(=O)C(Cl)(Cl)Cl)CO2 N1(C(c2c(C)cn(C)n2)=O)CCC2(C)CN(C(C3CN(C)C3)=O)CC12 C=CC(CC)CC(=O)N(CC(O)CN(C)C(c1cccc(OC)c1)=O)C C(=O)(CCCC(F)(F)F)NCC1CN(C(COCCCC#C)=O)CC(C)C1 C#CC(CNC(C1CC1C(C)NC(=O)C=C(C)C(C)C)=O)CC C(=O)(C1=CCS(=O)(=O)C1)NCC1CCN(C(Cc2cccc(C#N)c2)=O)C1 CC1CC(CNC(c2cccnc2F)=O)CN1C(c1cn(C2CCOC2)cn1)=O C1(NC(C(C)=C(C)C)=O)CCN(C)C12CCCN(C(C1(C(F)F)CC(O)C1)=O)C2 CCCCCCCC(=O)NC(C)C(C)NC(=O)C(C)OCCC(C)C Cc1cccc2cc(C(N3CC4CC(C3)C4NC(=O)CC(C)C)=O)oc12 Cc1cc(C(N)=O)ccc1NC(c1csc(-c2ccnn2C)n1)=O n1(CCC)nnnc1CNCC1(C(C)(C)C)CCCO1 C(=O)(CCN(OC)C(=O)c1ccsc1C#N)Nc1c(OC)cnnc1 C(=O)(C(N)C(=O)NCCCOc1ccncc1)OC c1(C(=O)NCCc2c(C(NOCC(C)(C)O)=O)c[nH]n2)cc2n(n1)CCO2 c1(C(N2C(CNC(c3c(C)cc(F)s3)=O)CCCC2)=O)cnn2c(N)ccnc12 C1(C(N(C(C)CNC(=O)CC2CC=CC2)CC)=O)OCCC1(C)C N12CCN(CC1=O)C(=O)C2.Cc1nc(CN(CC(C)C)CO)n[nH]1.C(C(C)(C)CO)N Cc1cc(F)ncc1-c1cn(CC2CN(C(c3cnc(C4CC4)s3)=O)C2)nn1 CC1c2ccccc2OC1CC(=O)N(C1CC(NC(c2ccc[nH]2)=O)C1)C N1(C(c2cncc(C#C)c2)=O)CC2(CCC(CNC(C3CCC(=C)CC3)=O)O2)C1 C1(C(C)NC(C2CC(N3CCCC3)C2)=O)CCN(C(C2(CF)CCC2)=O)C1 c1(C(N2CC(NC(CC(=O)OC)=O)C(C)C2)=O)cc(Cl)c(Br)cc1OC N1(CCC(=O)NC(CCOC)CNC(c2occc2C)=O)CCN(C)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CC(F)CC1CNC(=O)CCc1ccc(F)cc1 c1(C(N(CCNC(c2c(OC)n[nH]c2)=O)C2CC2)=O)n[nH]c2cc(C)ccc12 CC1C(C)S(=O)(=O)CCN1C(=O)NC(C1(C(F)(F)F)COC1)(C)C N1(C(C=CC=CCC)=O)CC(N2CCCC2)CC1OC(=O)NCC1CC1 C(CCSC)(C(=O)NC1CCC(C(N2CCC(CC3CC3)CC2)=O)CC1)OC(C)C C1(C(=O)NCC2(F)CCCN(C(=O)CN3CC4CC4C3)C2)CCCCC12CCC2 C1(C(=O)NCCCN(C(CCCN(C)C)=O)C2CC2)CC2COCC(C1)C2(F)F N1(C(C(C=C)(C)O)=O)CC2CCN(C(C3(O)CCCCCC3)=O)CC2C1 CCC(CCOC)N=c1nc2c(ncn2C)c(NCc2cc(Br)no2)[nH]1 N1(C(CCC)=O)CC(O)(CNC(C2(N3CCCC3)CC2)=O)C1 N1(C(C=C(C)c2ccsc2)=O)CCN(C(C2CCCSC2)=O)CC1C(C)(C)C CC(CCC(=O)N1CC(CNC(=O)Cc2cc[nH]n2)C(C)C1)S(C)(=O)=O c1(C(N2C(CO)CC(NC(C3C4CNC(=O)C34)=O)C2)=O)c[nH]c2ncccc12 C1(NC(C2CC(=C)C2)=O)CCC2CC1CN2C(C1CC(F)(F)C1)=O Cc1cc(C(=O)N(C)CC2CCC(NC(=O)C(C)OC(C)C)CC2)c(O)cc1F CC1CCC(NC(c2ccnc(OCCO)c2)=O)CN1C(=O)CCC(N)=O c1(C(C)=O)ccc(S(=O)(=O)NCc2cc3ccccc3n2C)c(C)c1 C1(NC(C(=O)Nc2c(C)nn(CC(F)(F)F)c2)=O)C2CCCCCC12 N1(C(CNC(CC)(C)C)=O)CCC(CNC(=O)CCC2CCCC2)C12CC2 c1(C(=O)NC2C(CC)N(C(=O)C(c3cncnc3)C)CC2)ncc(Br)cc1C CCC(C)C(O)C(C)C(=O)NCC1(C(=O)NCCCC(C)CO)CC1 c1(C(=O)NC2(C(=O)NCCC(CC)O)CC2)ccc(O)cc1 N1(C(C2ON=C(C)C2C)=O)CC2CC1CN2C(C12CC(C1)C(C#N)O2)=O c1(C(=O)NCC=C(C(=O)NC(C2CCOC2)CC)C)cnn(C)c1C#N C1(COC)(CNC(c2cccc(C)n2)=O)CCCN1C(c1csc(O)n1)=O C(=O)(C(C(C)C)NC(=O)C(F)(F)F)NCC(CN(C(CCC#C)=O)C1CC1)(C)C C1(C(=O)NCC2(OCC)CN(C(c3cc(Cl)ncc3N)=O)C2)CN2CCC1CC2 Cn1nnc(CNC(=O)CC(C2CC2)NC(c2ccnn2C(F)F)=O)n1 C(=O)(C1=CCCCO1)NCC(CC)NC(=O)Cc1ncc(-c2ccc(Cl)cc2)o1 C1(C2(O)CCOCC2)(C(=O)OC)CC1.c12cccc(c1)NC(=O)NC2 c1(C(C2CC2)OC)nnc(N2CCC(C3CCCO3)C2)n1CC.C1(=O)CCCO1 CCC(CC(C)C)C(=O)NCCCN1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 CN1C(=O)N2CC(NC(N3CCCCCC3CO)=O)CC2(C)C1=O c1(CNC(C2COC3(CCC3)C2)=O)ccc(C(F)(F)F)cc1Cl Cc1ncc(C=CC(N2CCCC(CCNC(=O)COC3(C)CCC3)C2)=O)s1 CC(=O)C(C)CC(C)C(=O)N1CC(C)C1C(=O)NCCc1cncs1 Cc1cn2nc(C(=O)NC34CCCC3N(C(C3CCCO3)=O)CC4)cc2c(=O)[nH]1 C1(C(=O)NCC2(F)CN(C(CN3CC(C)(OC)C3)=O)C2)CCC2CCC(=O)N12 N1(C(C(C)N(C(=O)C(=O)NOC)CCC)=O)CC(C)N(C)C(C)C1 N1(C(CCCOC(C)C)=O)CCN(C(C2CCOC2)=O)C2CCC12 Cc1ccc(C(N2CCCC(C(C)NC(C3(c4ncco4)CC3)=O)C2)=O)cc1C C1(NC(C2C(C=C)C2)=O)CCN(CCNC(C2CCC(C(F)(F)F)C2)=O)CC1 N1(C(C2(C#C)CC2)=O)CCCN(C(=O)CNNC(=O)Nc2ccc(F)cc2)C(C)C1.NC Cc1cc(NS(C)(=O)=O)ccc1C(N1CCCC1(C)CNC(=O)C(C)N(C)C)=O C1(C(=O)NCC2(O)CCC(C)(C)C2)CCN(C(=O)CCC(=O)C2CC2)CC1(C)C C1(CC(=O)NC)CN(C(c2cnco2)=O)CCN1C(=O)Cc1cncnc1 C=CCC(CC=C)C(=O)NCCC1CN(C(=O)C=CCCC)CC1C N1(C(c2nn(C)c(Cl)c2)=O)CC2CCC(NC(=O)CCOCC(F)F)(C2)C1 N1(CCNC(CC(C)C)=O)CCCN(C(=O)CSc2ccc(F)c(F)c2)CC1 C1(NC(C(CC)N(C)C)=O)CC(C(=O)NC2(N3CCOC3=O)CC2)C1(C)C Cc1cc(C)nc(N2CCC(CCNC(c3cnc(OC(C)C)cn3)=O)C2)n1 C1(C(=O)NCC(CNC(C2CCC(C)O2)=O)(C)F)CC2CCC1CC2 C(C(C(C)(C)C)NC(C1CCS1(=O)=O)=O)NC(c1ccc(COC)s1)=O CCCCC(C)(F)C(=O)NCCC1=CCN(C(=O)Cn2cccc(O)c2=O)CC1 Cc1cnc(C(=O)N(C(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)C)c(F)c1 C1(NCc2c(C)cc(C)[nH]2)CN(C(=O)CCOCC(=O)OC(C)C)CCC1(C)C C(C(=O)NOCC1CCOCC1)(C1CCC1)NC(CC1(C#N)CC1)=O N1(C(c2cc(C)[nH]c2)=O)CCC(CNC(=O)CC2(O)CCCCCC2)C(O)C1 c1(CC(N2CCCC(N(C(C=CC)=O)C)C2)=O)ccc(SC2CC3CC2C3)cc1 C1(C2CCN(C)CC2)(C(N2C(CNC(C3CC(C)NC(=O)C3)=O)CC2)=O)CC1 C(=O)(C(C)(C)C(O)C(C)C)N1CC2(CC(NC(CCc3ccc(C)s3)=O)C2)C1 c1(NCC(c2cn(C)nc2)O)ccc(S(=O)(=O)NCCC2CCC2)c(Cl)c1 N1(C(C2(C#C)CC2)=O)CC2CCCC2(NC(C2CC3OC2C2CC32)=O)C1 CC1(C)CN(CCO)CCN1C(c1cnc(-c2ccc(CO)o2)cn1)=O CC1(C(N2CCOCC2CNC(c2cnc(Cl)s2)=O)=O)CC(F)(F)C1 N1(C(c2ccc(OC)o2)=O)CC(NC(=O)CCc2conc2C)C(C2CC2)C1 c1(C(=O)NC2CN(C(C(CC)C)=O)C(C)C2)ccc(F)c2occc12 C1(CNC(C(OCC)OCC)=O)(NC(=O)C#CC(C)C)CCC(C)(C)C1 C(=O)(C1CC(=O)c2ccccc21)N1CC2C(CNC(=O)COCCF)(CCC2)C1 Cc1cccc2c1OC(C(=O)NC1CCCC3OCCC13)C2 c1(N(CC(C(C)C)O)C)ncc(S(=O)(=O)N2CCC(CO)C(F)(F)C2)cc1Cl c1(C(N(CCCNC(c2ccc(C(C)(C)C)cc2)=O)C)=O)cc(O)ccc1O CC1(C)CC2(CC2C(N2CCCCC(CNC(c3cccc(O)c3Cl)=O)C2)=O)C1 C#Cc1cc(F)c(C(=O)NCC(CNC(C2C=CCCC2)=O)CO)cc1F Cc1cnccc1C(=O)NCC1CCN1C(=O)CCc1cncc(Br)c1 C12(CNC(=O)Nc3cnn(Cc4ccccc4)c3)CCCCC1C2 C(CNc1cc(-n2ccc(C(=O)O)n2)ccn1)(C(F)(F)F)OC N1(CCC)CCC(NCC(c2ccc(F)cc2)NC(=O)NC2CC2)CC1 N1(C(C23CCN(C(C4CCC(OC)C4)=O)CC2C3)=O)CCN2C(=O)OCC2(C)C1 C1(NC(C(CC)SCc2ccccc2C)=O)CC2CCC(C1)S2(=O)=O c1(C(N(C)CC2CCCN(C(=O)CSCc3ncc[nH]3)C2)=O)cc(Cl)ncc1O C=CCCCC(C)(C)C(=O)NCC1CCN1C(c1cn(C)nc1-c1nccs1)=O C1(CCC)(NC(=O)C(C)C(C)(F)F)CCCN(C(c2cncnc2C(C)C)=O)C1 C(=O)(C(C)S(N)(=O)=O)N1CCN(C(C(C)(CSC)OC)=O)CC1.N1CCOCC1 C(=O)(CC(C)CC(C)C)N1CCCC(C(N(C)Cc2c(C)nn(C)c2)=O)C1 C1(CC)CCN(C(c2ccc(C(=O)NCC(=O)N(C)O)cc2)=O)C1C(=O)OC c1(CC=C)c(N2CC(N(C(=O)COCCN(S(C)(=O)=O)C)C)C2)nc(=N)[nH]c1C n1(CC)nc(C)cc1C(=O)NCC(C)C(=O)NC(C)C1CC1 c1(NC(C)C)cc(N2CCCC(CCNC(=O)CN(C)C)C2)ncn1 Cc1ccc2c(c1)CC(C(=O)N(CCN(C(=O)CCCCCO)C)C(C)C)O2 c1(C(=O)NC2C3CN(C(c4c(SC)nccn4)=O)C2C3)cc2ncccn2n1 C1(NC(C=CC(CC)C)=O)CC(C)CN(C(c2ccc(CS(C)(=O)=O)o2)=O)C1 n1(CC)nc(C)cc1C(=O)NCC1CC1C(=O)NC1(CC2CC2)CC1 C1(NC(C(C)N(CCC)C)=O)CC(Oc2ccccc2)C1(C)C OCC(CNC(c1nnnn1CCCF)(C1CC=CC1)C)CC1CC1 c1(CC)cnc(C(=O)N(CCC(C(C)C)NC(C2CCC=CCC2)=O)C)nc1 C(c1ccc2occc2c1)=CC(=O)NC1CC(C)(NC(c2cnc[nH]2)=O)C1 N1(C(CC(CC)SC)=O)CCC2CN(C(c3nc4c(s3)COCC4)=O)CC12 C1(CC)C(NC(=O)CC2COCC(C)O2)CCCN1C(C1CC(=O)NC(C)C1)=O Cc1nc(C(=O)NC2(CNC(c3ccc(Cl)cc3)=O)CCCC2)n(C)n1 N1(C(C2(CCC)CCC2)=O)CCC(F)(CNC(=O)CC2CC=CCC2)CC1 N1(C(C2(C)CC(NC(C(C)c3cc[nH]n3)=O)C2)=O)CCOCC(C2CC2)C1 CC(CN=c1ccn2nccc2[nH]1)NC(c1coc(S(C)(=O)=O)c1)=O C(=O)(CC(C)(C)N(C)C(C1CCCO1)=O)NC(C)CCn1cncn1 C(=O)(C1=CC(O)C(NC(=O)C(C(C)(C)C)OC)C1)NCC(CC)(C)C N1(C(c2c(C)scn2)=O)CC2CC1C2C(N1CCC(n2cccn2)C1)=O Cc1cccc2c1OC(C(=O)NCC13CC(NC(C4CC45CC5)=O)(C1)C3)C2 CC(C(=O)N1CCC(NC(=O)CN2CC3CC3C2)C1(C)C)C(F)(F)F CCCCC(C(=O)NC(C)CNC(=O)CCC1(C)CC1)C(C)C N1(C(c2cc(SCC)sc2)=O)CCC(N(C(=O)CCC2CCCN2C)CC)CC1 CC(CC(=O)NCC(C)(C)CNC(C1CC(n2cccn2)C1)=O)n1cccn1 C1(C(=O)NCCC(C)N(C(=O)Cc2ccc(Br)nc2)C)CCC2(CCC2)O1 N1(C(=O)ON2CC(CC)OCC2)CCN(Cc2cccc(C(=O)OC)c2)C(C)C1 c1(C(N2CC=C(CNC(C(C(C)OC)O)=O)CC2)=O)cnc2ccoc2c1 Cc1nc(N)cnc1C(N1CCC(NC(=O)CC2CCCOC2)C1)=O S(=O)(=O)(c1cc(C(N2CC(CCNC(C3CCCC3)=O)C2)=O)ccc1OC)NC C1(C(=O)NC2C(CNC(c3cnns3)=O)CCC2)CCCC2CCCN12 C(=O)(C(CCCC=C)NC(c1ccc(F)cc1F)=O)NC(C#CC#C)(C)C c1(CC(=O)NC(C)CCN(C)C(C2CCC(=O)N2)=O)cnccc1C(F)(F)F C(=O)(CN=c1cc[nH]cc1)ONC(C12CC(CO)(CN1CCC(C)O)C2)=O N1(C(c2cc(C)c(C)s2)=O)CCN(C(C2CN(C3CCOC3)C2)=O)CC1C1CC1 c1(CCC)ccc(N)c(C(N2CCCC(NC(C3(F)CC3C)=O)CC2)=O)c1 c1(OC(C#C)=O)cc(CN2CCN(C(C)=O)C(CC#N)C2)ccc1Cl Cc1ccnc(C)c1C(=O)NCC(Cc1ccccc1)NC(=O)CN(C)C1CC1 C(=O)(C(C)CCC(C)(C)C)NCC(CC)(CC)NC(=O)C#CC1(C)COC1 c1(C(N(C)CC2N(C(c3c(C)cc(CC)o3)=O)CCCC2)=O)cnc(C)c(C)c1 c1(C(N(CC(C)NC(C(C2CCC2)NC(C)=O)=O)C)=O)ccc(F)c(C)c1N c1(C(N2CC(N(C(C=C(C)CCc3ccccc3)=O)C)C2)=O)nscc1N C(c1ccccc1Cl)=C(C)C(=O)NCCNC(c1ccc(SC(C)C)nc1O)=O C(C(=O)NOCC(=C)C)(C(C)(C)O)NC(C(C)OCC#C)=O C1(F)(C(=O)NCc2ncc(C)s2)CCN(C(=O)C(C)CC2CCCC2)CC1 c1(C(=O)NC2CN(C(C=C(CC)CC)=O)CC(O)C2)cc2c(Cl)nccc2s1 c1(C(N2CCC(N3CCN(C(c4c(C)coc4)=O)CC3)C2)=O)cc(N)cc(O)n1 c1(CC(N2CC(C3(NC(CC#N)=O)CC3)C2)=O)c(Br)ccc(F)c1F N1(C(c2ccc(C(N)=O)[nH]2)=O)CC2CCC1C(NC(c1ccccc1Cl)=O)C2 c1(NC(C2CNC2)C)cc(N2CCCCCC2)nc(F)c1 c1(C=C(C(=O)NCC(C2CC2)NC(=O)CC(F)(F)Cl)F)ccc(F)cc1F c1(OC)ccc(C(=O)N(C2CN(C(c3n[nH]cc3Cl)=O)CC2F)C)n2nccc12 C(=O)(C(C(C)C1CCC1)N(c1ccc(Cl)cc1)CCC#N)NCC(=C)C N1(C(CC2CC(C)C2)=O)C2CCC1CC(N(C)C(c1cc(F)ccc1F)=O)C2 C1(C(N(CCOCC)C)=O)CCC(C)N1C(c1cnn(C(C)C)n1)=O CC1=C(C)CC(C(N2CCC(NC(=O)CCSc3n[nH]c(C)n3)CC2C)=O)CC1 Cc1cc(N2CCC3CCC(C2)N3)c(Br)cc1[N+](=O)[O-] C(CCC(C(=O)N1CC2CC1CS2=O)NC(=O)Cc1cnns1)OC Cc1cc(N2CCC(C3CCCC3)CC2)nc(=NCCC2CN(C)CCO2)[nH]1 Cc1cc(N)ccc1C(=O)NCC1(CC(=O)NC2CC2CN(C)C)CC1 C(=O)(C#CC1CCCO1)N1C2C(NC(c3c(SC)nn(C)c3)=O)C(C2)C1 c1(N(CC(O)COC)Cc2cc(OC)nc(C)c2)ncc2ncn(C)c2n1 c1(C(=O)NCC2N(C(C(C3CCOCC3)OC)=O)CCC2)cnc2nccn2c1 c1(C(=O)NC2C(NC(Cc3nnc(C)o3)=O)COC2)nc(Cl)sc1Br CC1CCN(C(=O)C2=NNC(=O)C2)CC1N(C(=O)CSCc1ccc(F)cc1)C C(=O)(C(F)Cc1ccccc1)N(CCCNC(=O)CCc1cscn1)CCO C=C(CNC(c1csc(CO)n1)=O)CCNC(C1CCC2CC12)=O C(=O)(CC(C)(C)CC(F)F)N1CCC(CC(C)NC(C2CN(C)C2)=O)CC1 c1(C(=O)NC(CN(C(C2C(C(C)C)CCO2)=O)C)(C)C)occ2c1CCC2 c1(-n2cc(CNC(N3CC(OC)C(F)C3)=O)nn2)nc2cc(Cl)ccc2s1 Cc1cc(-n2ncc(C(=O)NCCn3cc(-c4c[nH]nc4F)nn3)n2)cc(C)c1 c1(CC)cccc(CC)c1CC(=O)NC1(CO)CN(C(=O)Cc2cnoc2)C1 CC(O)C(C)C(=O)N(CCCNC(C1(c2ccno2)CC1)=O)C1CC1 CC(C)C(C)(O)CNC(=O)C(Cc1cn[nH]c1)NC(=O)Cc1cnns1 c1(C(C(=O)N(C(CC(=O)OCC)C2CC2)C)F)cccc(F)c1 C1(NC(CCNC(CCC2CCC2)=O)=O)CCC(C)N(C(=O)CC2CCSC2)C1.CO N1(Cc2n(C(c3ccc(C)nn3)C(=O)NC)ccn2)CCOC(C)(C)C1C N1C(=NCCCCCl)N2CCC(C2)SCCC1.c1(SCC)ccccc1.N(CC)(CC)CC C(=O)(C1=Cc2ccccc2C1)NC1C=CCC(C(=O)NC(CC)(CC)CC)C1 C12(CNC(CC(C=C)CCC)=O)CC(NC(c3nc(=O)n(C)[nH]3)=O)(C1)C(C)(C)O2 N1(C(C=CCCC)=O)CCCCC1CC(=O)NC1(CF)CC(=O)C1 c1(C(N(CCCNC(C2C(C=C)CC2)=O)C)=O)sc(=N)[nH]c1C C#CCCCC(=O)N(CCCOCCNC(C1CCOC(C)C1)=O)C n1(CCN=C(NCc2c(F)cncc2)NCC2(F)CCC2)cnc2cccnc12 N1(C(C=CCC)=O)CCN(C(c2ccc(Cl)cc2Cl)=O)CC1COC C(=O)(C(CNC(=O)CC1CCN(C)CC1)C(C)C)NC(CC)C(C)C CCCCCCC(C)C(=O)N1CC(COC)(NC(=O)C(C)(F)c2ccon2)C1 C1(C(=O)NCC(C)(C)NC(c2ccc(=N)[nH]c2)=O)CCCC1(F)F N1(C(Cc2c(C)ncs2)=O)CCC2(NC(c3cnc(O)cc3C)=O)CC2C1 CN1CCN2C(C1)C2=O.c1(CNC(C2CC3CCC(C2)O3)=O)ncc(F)cc1F C(=O)(C(C)(C)C(F)(F)F)NC(CNC(C1CC2(CC(OC)C2)C1)=O)CO C1CC[Si](C)(C)CN1.C(C(O)(C(F)(F)F)c1ccc(Cl)cc1)C1C(C)CCC1 N1(C(C2COCC(C)O2)=O)CC(C)(C)C(NC(c2ccccc2Cl)=O)C(C)(C)C1 N1(C(c2cc(C)oc2)=O)CCC2(CC1)CCN(C(=O)CC1CCCC1O)CC2 C1(NC(c2c(C)c[nH]n2)=O)CC2CC1N(C(=O)Cc1ccc(C(=O)OC)cc1)C2 N1(C(c2cc(CC)c(C)s2)=O)CCCCC(NC(c2cc(C)ccn2)=O)C1 CC(CC(=O)NCC1(C(=O)NCc2cncc(F)c2)CCCC1)C(F)F C(C(C)(C)CC(=O)NCC1CCN(C(C2CC(=O)N2)=O)CC1C)OC C1(C(N2C(C)CC(CNC(CNC(=O)OC)=O)C2)=O)CC2(CCCCC2)C1 c1(C(N2CC(NC(CSCCCC)=O)C(C)C2)=O)noc2c(F)cccc12 c1(OC)cc(C(=O)NCCCNC(c2cnn(C)c2)=O)cc2cccnc12 CC1CCN(C(=O)CN(c2ccccc2)Cc2nccn2C(C)(C)C)C1 C1(NC(C2(CCCC(=O)NCC3(C(C)C)CC3)CCC2)=O)CCC(O)CC1 C12(NC(C(CCC)NC(=O)COCCCC(C)C)=O)CC(CC(C)O1)C2 N1(C(C2CC(C)(C)C2)=O)CC2CCCC2(NC(c2cc3n(n2)CCO3)=O)C1 N12CCn3ncc(c3C1)C2=O.N1(Cc2n(C(C)C)ncc2)CCNC2(CCC2)C1 CC1C(NC(=O)C2CC2)CCCN1C(c1ccc(C(F)F)s1)=O C(=O)(C(F)C(C)(F)F)N1CC(N(C)CN2CCCC2)CCC1 c1(C(N(C2CCN(C(C3CCCS3)=O)C2)CC)=O)ccc(SC)s1 N1(C(C2(C#C)CCCC2)=O)CCC(F)(CNC(=O)COc2ccc(Cl)nc2)CC1 c1(NC(=O)COC2CCC2)ccc(CCN(C)C)cc1.C12CC1C(=O)N2 C1(CNC(C(CC)NC(c2ccco2)=O)=O)(CCl)CC(F)(F)C1 C(C(=O)NC(C(=O)N(C)Cc1ccco1)c1ccco1)(C1CC1)SC c1(C(N2CC(NC(c3c(C)ccnc3)=O)C(F)C2)=O)cccc2c1CCCC2 N1(CCS(=O)(=O)NCc2c(C)occ2)C(=O)NC(C)C1=O N1(C(c2cc(N)cc(O)n2)=O)CCC2CN(C(=O)C(=O)NCC(F)F)CC2C1 c1(C(C(C)C)N(C(=O)C(O)CC2CCNCC2)C)ccccc1 c1(CNC(N2CCCC2CNc2ncccc2F)=O)ccncc1C(F)(F)F C1(C(=O)NCCCCCCN2CCNCC2)CCCC2(CC2)C1 C1(NC(=O)NC2(C(N(C3(C)CC3)C)=O)CC(F)(F)C2)CC12CCCCC2 N1(C(c2cccc(Cl)c2Cl)C)CCC(F)(F)C(CNc2c(C#N)cnn2C)C1 C(=O)(C1=CC2(CN(C(=O)CCC3CCCO3)C2)OC1)N1CC(C)(C(C)C)OCC1 c1(C(=O)NC(C(=O)N2C(COC)CC2)CC2CCC2)ccc(C)nc1 O=C(CN=c1cc[nH]cc1)NC1CC2CC1CC2C(=O)NCc1cccnc1O Cc1cc(N2CC3CC(NC(=O)CNS(=O)(=O)N(C)C)C3C2)nc(C(C)C)n1 c1(NCCC(=O)NCC)ncc(C)cc1S(=O)(=O)NC1CC(OC)C12CCC2 CC(C)CCCCCCNC(C1(N(C(=O)C=Cc2ccccc2)C2CC2)CCC1)=O c1(OC)cccc(C#N)c1C(=O)Nc1cccc(-c2cccc(F)c2N(C)C)n1 C(=O)(C(C)CCCC(C)C)NC(CC(C)C)CC(=O)NCCN(C)C Cc1cc(O)c(F)cc1N=c1[nH]c(N(C)CC2CCOC2C)nc2c1CCCC2 Cc1cc(C)c(-c2cn(CCCN(C(=O)CC3CCSC3)C)nn2)cn1 N(C(=NCC1COC2(CCCCC2)O1)N1CCC(F)(F)C2(CCC2)C1)CCO C(c1ccc2c(c1)CCO2)=CC(=O)NCC(CNC(c1cc(C)c(O)cc1)=O)F C#Cc1cc(C(=O)NC2COCCC2NC(=O)C(CC=C)C(C)C)ccc1C N1(C(C(CC(N)=O)NC(=O)CN2CCCCC2)=O)CCc2nncn2CC1 N(C1c2ccccc2CCC1C)C(C(=O)Nc1cc(C)nc(C)c1)=O C(N=c1[nH]c(=N)[nH]c(=NC2CC(OCCO)C2)[nH]1)c1c(CCC)nns1 CS(=O)(=O)CC(=O)N1CC(NC(C2COCCN2C(C2CCC2)=O)=O)C(O)C1 c1(OC)ccc(C2CCN(C(=O)CSC)CC2)cc1OC C12(CC=CC1)C(=O)CCC1CC1C(=O)NC2.N1(OC)CC(N2CC(O)C2)C1 N1(C(Cc2c(C)nsc2)=O)C2CCCC1CN(C(C1CC(=O)CCO1)=O)C2 N1(C(C(CCNC(=O)CC(C)(F)F)OC)=O)CCC(O)(C2CC2)CC1 C(=O)(CCCN=c1nccc[nH]1)NCC1(O)CN(C(C=CS(C)=O)=O)C1 c1(C(N(CCOC)CCNC(=O)C(C2CCCCC2)O)=O)noc2c1COCC2 N(C(=NCC(C(C)C)C(C)C)NCC1CCCO1)CC1(OCC)CCCC1 c1(NCC(c2nccs2)C)[nH]c(=NCc2conc2Br)nc2scnc12 CN1CCN(C(=O)C2=CCCSC2)C(C(=O)NCC2COCCO2)C1 c1(NC(CCC)CCCNC(c2csc(C)n2)=O)nc(Cl)nc2c1cnn2C Cc1ccc2c(=NCC3CCS(=O)(=O)CC3)[nH]c(=NC(C)c3conc3Br)[nH]c2c1 c1(NC(C2N(Cc3ccn(C)n3)CC(F)C2)=O)c(Cl)cc(Br)cc1[N+](=O)[O-] N1(C(c2ccc(C(C)=O)s2)=O)CCCC12CCN(C(=O)CCCC(N)=O)C2 CC(C)C(C(=O)NCCC(C)CCNC(=O)CC1CC2(CCC2)C1)NC=O c1(C(N2C(C)CC(CNC(CNC(=O)OC)=O)C2)=O)cc2nccnc2cc1F N1(C(C(CC)N(C)C)=O)CC(NC(=O)Cc2c(Cl)cccc2Cl)CC2(CCC2)C1 N1(C(CC(C)(C)C)=O)CC(NC(c2ncc3[nH]ncc3n2)=O)C2CCCC2C1 C(c1cccnc1)=C(C(=O)NC1CCN(C(C(C)(F)c2ccccc2)=O)C1)F Cn1c(=O)n(CC(=O)NC(CNC(=O)C(O)CC[S+](C)C)CO)c2ccccc12 n1(C(C)C)ncc(C(=O)N(C2CCC(NC(=O)C(C3CC3)C3CC3)CC2)C)c1N c1(OCC)cc(C(=O)N(CCCNC(=O)CC2CCC2=O)C2CC2)ccn1 C1(O)(CCNC(C=CSC)=O)CCN(C(=O)CS(=O)(=O)Nc2ccccc2)C1 C1(C(=O)NC(CC)CC(=O)OC)(NC(=O)CN(C)C)CCC(C)(C)C1 N1(C(c2c(C)nns2)=O)CCC(O)(CC(=O)NCc2cccc(O)c2C)CC1 C1(CN(C2(C(=O)NCC3CCOC3)CC2)C)C2CC=CCC12 c1(-c2cc(C(=O)NCC=CCNC(CC3C(C)C3)=O)on2)cccc(Cl)c1 C1(CC(=O)NCC2CC(OCC(=O)N(C(CC)C)CC)C2)CCCC1C c1(-c2nc(CCCCC)nn2C2CCS(=O)(=O)C2)cc([N+](=O)[O-])c2nsnc2c1 C1(C(=O)Nc2ccc(OC(C)=O)nc2)(OC)CCCN(C(=O)CCOC(C)=O)C1 Fc1cc(NCCCC2COCCOC2)c(F)cc1Cl C(=O)(C1=C(C)N(C)c2ncnn2C1C)N(CC(CNC(C(C)SC)=O)O)C N1(C(C(F)OC)=O)CC(NC(=O)CCc2cc(C)on2)C(C)C1 C(=O)(C1=C(C)OCC1)NC(c1ncccn1)CC.c12ccc(cn1)CNC2=O c1(C(=O)NC2CC(CNC(C3(c4ccc(OC)nc4)CC3)=O)C2)cnc2n1CCS2 Cn1ccc2cc(-c3ccnc(N)c3)cnc12.S(=O)(=O)(c1ccncc1)N1CCC1 c1(C(C)=O)cc(CC(C)=CC(=O)NCCCNC(C2(C)CCOC2C)=O)c(C)o1 c1(CCN2CCC(C(C)NC(=O)C3=CCCC3)CC2)cccc(Cl)c1Cl S(=O)(=O)(c1cccnc1N(C)Cc1ccccc1Br)NC(C)CCOC(F)(F)F C12(CC(N3CC(NC(C=CCOCCOC)=O)C(O)C3)=O)CCCN1CCC2 C(C)(N=c1[nH]c(=NCCF)[nH]c2c1CSC2)c1n(C(C)C)ncn1 Cn1cc(CCC(=O)NCC2(C(=O)N(CC(F)(F)F)CCO)CCCC2)cn1 C1(NC(c2cc3ncccc3[nH]2)=O)CCC12CCN(C(=O)CSC1CC1)CC2 N1(C(c2cccc(SC)c2Cl)=O)CCC2CN(C(=O)C3=NOC(C)C3C)CC12 c1(C(N2CCCC(C)(CNC(C3CCCCC3O)=O)C2)=O)[nH]nc2ncccc12 C12(CF)CC(CN3CCC(OC4CCC4)CC3)(CO1)C2 C12(C(=O)NCCOC3CN(C(c4c(CC)con4)=O)C3)CCCC(=O)N1CCC2 CCC(C)CC(=O)NCC(C1CCCN1C(=O)CCc1cccc(OC)n1)(C)C C1(CNC(CCC#C)=O)CN(C(c2ccc(Br)c(N)c2)=O)CCC1(C)C N1(C(C(C)c2cc[nH]n2)=O)CC2COCC2(C(=O)N(C2CC2)CC2CC2)C1 C(=O)(C(O)P(C)(C)=O)NC(c1ccccc1)CNC(CCC(=O)OCC)=O C1(C(=O)NCC2(CN(C(=O)CC(C)(C)O)C)CC2)CCC2(CCC2)CC1 Cc1nn2ncccc2c1C(=O)NC1CCCC1CNC(=O)Cc1ccsc1C CC(C)CCCCC(=O)N1CCCC1(C)CCC(=O)NC1(C)CC1(C)C c1(C(N2CCC3(NC(=O)CCNC(=O)CO)C(C2)C3)=O)cn2cccnc2n1 c1(NC(C(=O)N(CC(C)C)Cc2c(C)c(F)ccc2)=O)cnn2ccc(O)nc12 C1(C(=O)NCC2(C(N)=O)CN(C(C3CCCC3)=O)C2)CC12CCCOC2 C(=O)(C1CCCc2nccn21)NC1CC2(CN(C(C3CC=C(C)CC3)=O)C2)C1 c1(C(=O)NCC(C)(C(C)C)NC(C(CC)F)=O)c(F)cncc1Cl C1(NC(c2ccn(CC)n2)=O)CCCCC1CNC(=O)CC(C)c1ccncc1 C1(NC(c2cnc(C3CC3)nc2O)=O)CN(C(C2CCCC2)=O)CCC1CO CCC(C#N)C(=O)NC(C)C(CO)NC(c1cocc1C)=O C1(C(N2CCC(NC(c3cc(CC)no3)=O)C(CO)C2)=O)CCS(=O)(=O)C1(C)C C1(N(C)C(C2SCCS2)=O)CC2CC1N(C(c1cc(F)cc(Cl)c1)=O)C2 C1(NC(c2ccc(N(C)C)cc2)=O)CCN(C(c2cc(C(F)F)no2)=O)CC1O N1(C(=O)CCc2ccsc2)CCOCC(C(N2CCOC3CC23)=O)C1 C(=O)(CCN=c1ccc(S(=O)(=O)NCC(C)C2CCC2)c[nH]1)NC CC12CCCC1CN(C(C1(NC(c3c[nH]c(=O)cn3)=O)CCOCC1)=O)C2 c1(C(N2CC(NC(C(C(C)OC)O)=O)(CF)C2)=O)ccc2nnnn2c1 C1(C)(C(=O)NC2CN(C(CSc3cccc(C)c3)=O)C2)CCCCC1C Cc1cc(=O)c(C(=O)NCC(C)(C)NC(=O)Cn2cccn2)cn1C1CC1 c1(C(C(=O)NC(C)C)N(C)C(c2cccc(Cl)c2)C)sc(Cl)cc1Cl c1(NC(C2(C)CCN(C(C(C)NC=O)=O)C2)=O)c(Cl)cc([N+](=O)[O-])cc1Br c1(C(CC)C)nc(CC2COC(=O)C2)n(-c2c(C)noc2C)n1 C1(NC(c2c(CC)non2)=O)CC2CCC(C1)N2C(C12CCCC(C1)OC2)=O c1(-c2cc(C)c(OC(C)C)nc2)cnc2[nH]c(C(N3CCC(O)C3)=O)cc2c1 CCC(C)C(CC(=O)NCC(c1ccccc1)O)NC(C1CC(C(C)C)C1)=O CC(C)(C)C(=O)NCC1CC1.C1(=O)CC(=O)NCCCN1 c1(C(=O)NCCCC(C)NC(=O)CCNC(=O)CO)cc(Cl)ccn1 c1(C(=O)NC2C(C(=O)NC3C(OC)COC3)C2(C)C)ccccc1O c1(C2(C(N(CCNC(CC(=O)OCCC(C)C)=O)C)=O)CC2)ccc(F)c(Cl)c1 C#CCC(C(N)=O)NC(=O)C(C(C)C)NC(c1ccc(CO)nc1)=O C(=O)(C(F)C(F)(F)F)N1CC(CNC(c2csnn2)=O)OCC1 C(CCOC)(C(N)=O)NC(C1CCN(C(c2c(CC)nns2)=O)C1)=O C(C(C)(C)C)C1(NC(N2CCCC2)=O)CC1.C(=O)(C(C)(C)C1CCCO1)NC(C)C C=C1CC2(C1)CC(C(=O)NCC(CNC(c1ccsc1C)=O)C(F)(F)F)C2 Cc1oc(C#N)cc1C(N1CC(NC(c2cnc(C(F)(F)F)s2)=O)C2(CC2)C1)=O C1(NC(C(CC#C)(C)C)=O)CC2(CCN(C(C3CCC3C#N)=O)C2)C1 C1(C(N)=O)(OC)CN(C(c2ncoc2CNC(=O)C(c2cncn2C)O)=O)C1 N1(C(CC2CCCC(C)C2)=O)CC2CCC1C(CNC(C1CC1C)=O)C2 c1(NC(C2N(Cc3scc(C)c3)CC(F)C2)=O)cccc(C)c1O C(C(=O)NC1CCCC1C(C)C)(C(C)O)NC(C=CCOC)=O N1(C(c2c(OCCC)cccn2)=O)CCC(CNC(C2CCCS2)=O)C1(C)C C(=O)(C1=CC2C=CC(C1)C2)N(CCC(=O)N(C1CNC(=O)C12CC2)C)CC#C C(=O)(CCCCCC(C)=O)N(CCC(C)NC(C(COC)OC)=O)C C1(C(=O)NC(C)CNC(c2cc(Cl)n(C)n2)=O)CCN(CCO)C(=O)C1 N1(Cc2ccc(C)c(O)c2)CCN(C(c2cc([N+](=O)[O-])cs2)=O)C(C#N)C1 Cc1nc2cc(C(=O)NC(C)(CNC(=O)C(C)(O)C3CC3)C(C)C)ccc2s1 C1(CNC(CCCC#C)=O)CN(C(=O)C(F)=CC2CC2)CC1(F)F O(NC(=O)CC(CC)C(CC(=O)N)C)CCCCC#C.S(C)CC C(C(Cc1ccccc1)C(F)(F)F)NC(=O)NC1CCCCC1.C1C(=O)N1 c1(OC)ncc(Br)cc1CC(=O)NCC(C)NC(C1CC(F)C1)=O c1(NC(C2CCC(O)(c3cccc(F)c3)CC2)=O)cccc(Cl)c1-n1ccnc1 c1(C(=O)OC(CC(C)C)C(=O)N(C)C)n[nH]c2c1CCC(C)(C)C2 CCC(CCCC(=O)NC1(C(F)F)CC(C(N)=O)C1)NC(c1cn[nH]c1)=O c1(SC)cc(C(N2CCC2CNC(C2CCCC23CCC3)=O)=O)ccc1F C(=O)(C1CCCn2nccc21)NCC1CCCCN(C(C(F)=CCC)=O)C1 Cc1noc(C)c1C(c1nnnn1CC(F)F)NC1CCC(CCO)CC1 c1(OC)ccc(CC(N2CCCC2CNC(=O)C(C)(C)CSC)=O)cc1F C(CN=c1nc(CC)[nH]s1)(C1CCC(CC)CC1)NC(C(CC)NC(C)=O)=O C1(CC(=O)N(CCNC(CCOCCOCC)=O)C)CCCS(=O)(=O)C1 N1(C(c2cc(C(=O)OC)cc(Br)c2)C(=O)NCCC#N)Cc2c[nH]nc2C(C)C1 c1(C(=O)NCC(CC=C)NC(c2ccncc2F)=O)n[nH]c(C)c1C(F)(F)F N12CCC(C1)NC2=O.C12CN(C1)C(=O)C(=O)NC2C.C1(CN)CC1.CN N1(C(c2c(SC)snn2)=O)CC(CNC(c2ccc(C(F)F)cc2)=O)CC1C N1(C(C(Br)=C(C)C)=O)CC2(C1)CN(C(C1CCC(=O)C(C)C1)=O)C2 N1(C(c2cn(C)nn2)=O)CCC2(CCCC2CNC(c2ccc(N)cn2)=O)CC1 CC(CCCCCO)NC(c1csc(CNC(=O)CC2(C)CCCCC2)c1)=O Cc1cccc(OCC(C)N(C(C2CCC(C)C2)C(=O)NCC(C)C)C)c1 C1(C(N2CC(CCNC(C(C)OCCOCC)=O)C2)=O)CCn2nnnc2C1 CCC(C)(C(=O)N(C)CC1CCCN(C(c2ccc(COC)o2)=O)C1)C(N)=O CC(C)(C)C(O)CCC(=O)NC1CN(C(=O)CC2(CO)CCC2)CC2(CC2)C1 c1(CNC2CCC(C(=O)NCC3CCC(CO)CC3)C2)c(O)cc(O)cc1O N1(C(C2COCCO2)C(=O)NCCC#N)CCC(F)(c2ccccc2)C1 C#CCC(C(=O)NC1(c2noc(C)n2)CC1)NC(=O)C1CC1 CC(C)C(C)CC(=O)N1CCC(CNC(=O)CSc2cn[nH]c2)C12CC2 CC1CCc2[nH]nc(C(N3CCOC(CN(C)C(C45CC(C4)C5)=O)C3)=O)c2C1 C1(NC(N2CCN(C3C(=O)NC(=O)C3)CC2)=O)C(F)CC12CCC2 Cc1ncc(C(=O)NCC2CCN(C(c3c(Cl)cnn3C3CCCC3)=O)C2)n1C c1(OC)ccc(CCNC(N2CCC(CO)CC2C)=O)cc1Br c1(NC(C2(C)CCCN2)=O)nc2ccc(Cl)cc2s1.N12CCCC1C2=O C(C)(C(C(=O)N1C(=O)NC(C)(C)C1=O)C(C)C)OC(Cc1c(C)noc1C)=O c1(OC)cc(F)c(-c2cc(C(N3CC4CCCCC4C3)=O)no2)cc1OC C(=O)(C(CCS(C)(=O)=O)NC(=O)CC(=O)Nc1cccc(Br)c1)OCC N1(C(C(C)OC)=O)CCN(C2CCCN(C(c3ccnn3C(C)C)=O)C2)C(=O)C1 C1(CC)CN(C(c2ocnc2C2CC2)=O)CCN1C(=O)C=Cc1ccn(C)c1 c1(OC)cc(C)c(NC(c2nnnn2C2CCOC2)c2cc[nH]n2)cc1F N1(C(=O)CN2CCSCC2)CC2CN(C(c3ccccc3Cl)=O)CC2C1 C1(NC(c2ccco2)=O)CC2CCC1(CNC(c1cc(C(F)F)ccc1O)=O)C2 CN1C(=O)N2CCC(C(=O)NC3CN(C(=O)C=CBr)CC3O)C1C2 c1(C(=O)NCCCCCN(C(=O)Cc2cnoc2)C)ccc(Cl)c(F)c1 C1(O)(CNC(C(COCC)C)=O)CCCN(C(=O)Cc2cccc(F)c2)C1 C1(C(C)NC(CCc2ccc(C)s2)=O)CCCCN1C(=O)C=Cc1cnc[nH]1 CC(CN=c1[nH]c2ccc(S(=O)(=O)NCC3CC(=O)N(C)C3)cc2s1)OCCO N1(C(c2nc(CC)oc2C)=O)CCC(NC(=O)C=Cc2ccc(C)o2)C12CCC2 N1(C(c2sccc2C(F)F)=O)CCC(C(F)F)(CNC(C23COCC2C3)=O)C1 CC1=C(C(=O)NC(c2ccco2)CO)C(C)n2ncnc2N1C C(=O)(CCCSC)N(C(CNC(c1cnn(C)n1)=O)Cc1ccccc1)CC c1(NC(C2CCN(c3nccc(C)c3)CC2)=O)cc(C)c(F)cn1 Cc1nc2c(o1)CCN(C(c1ccnn1C)C(=O)NCc1ccccc1Br)C2 c1(OC)cccc(C(O)CNC(C2CC(=O)N(Cc3ccccc3)C2)=O)c1 CCC(C)(CNC(C1CC(=O)N(C)C1)=O)C(=O)NCc1nc(COC)n[nH]1 c1(C(=O)NC2CC(NC(c3n[nH]c(C)c3Br)=O)C2)ccc(Cl)cc1C#N c1(CC(=O)N(C)CC2OCCN(C(C3(COC)CC3)=O)C2)ccc(C#N)cc1 c1(NC(=O)CC(F)C(C)C)ccc(C#N)cc1O.Cc1oc(C(=O)NCC)nc1 CCC1=NOC(C(=O)NCC(C23CCC(CC2)C3)NC(c2nn(C)cc2C)=O)C1 c1(C(N2CC3C(NC(=O)CN4CCCC4=O)(C3)C2)=O)cnn2ccncc12 c1(OC)cccc(C(C)(C)C(=O)NCC(C)CN(C(=O)CC2CN(C)C2)C)c1 CCC(CC(=O)N(CC(C)C(C)C)C)NC(c1cn(C)nc1C)=O N1(C(c2cccc(OC)n2)C(=O)NC2CCC2)CCc2c(ccnc2Cl)C1 C1(NC(C2CC(OC)C2)=O)CC(NC(=O)CCc2cccnc2Cl)CC1O Cc1sc(C(=O)NCCOCCCNC(=O)C(F)(F)C2CCCC2)cc1[N+](=O)[O-] c1(OC)ccc(C)cc1CC(=O)NC1C2CN(Cc3cc(C)ccc3I)CC12 Cc1cc(F)c(C(N2CC(CCNC(c3coc(C4CCC4)n3)=O)C2)=O)c(Cl)c1 c1(C(=O)NC2CN(C(c3c(CC)occ3C)=O)CC2C)ccc([N+](=O)[O-])c(C)c1 C1(C)(NC(CCCCSC)=O)CCCCC1C(N1CC2CC1CS2=O)=O c1(NC(N2CC(C(=O)OCC)C2)=O)noc2cc(-c3cccc(C#N)c3)ccc12 C(N=c1nc(N2CCC3(CCOC3)C2)c2c([nH]1)CCOC2)c1n(C(C)C)ncn1 c1(CC)c(C(=O)NC23CC2CN(C(c2snnc2C)=O)C3)csc1C c1(CCC(=O)NCCC2CN(C(C(C)n3ccnc3)=O)C2)cccnc1 c1(C(=O)NCC(CNC(C(C)CSc2ccccc2)=O)O)cc(N)c(F)cn1 N1(C(CCNC(=O)OC)=O)CCCCC(NC(=O)CC2C(=O)ON=C2C)C1 N(CCCN=O)(C(CCNC)N1C(CCSC)C1=O)CC C=CCCCC(C(=O)NCc1c(C)nn(C)c1C)NC(c1ccsn1)=O C1(CNC(C(C)OCCCC)=O)OCCC1C(=O)NC1(CN(C)C)CCCC1 C(=O)(C1COc2ccc(Cl)cc21)N1CC(NC(C(C)n2ccnc2)=O)C1 C(CC(C(=O)NCCC(=O)NC1CC1)NC(C1(C#N)CCCO1)=O)N(C)C C1(C(=O)NCC2CCCN(C(c3c(C)ncn3C)=O)C2)C(C)OC(C)C1C c1(C(=O)NCC(CC)NC(C2CC2c2ccccc2OC)=O)cccc2nccn12 Cn1nc2c(c1C(=O)NCC1COCCN1C(c1cc(F)ccc1O)=O)CCC2 c1(C(=O)NC(C)(C)CNC(C2CCCCC2O)=O)ccc(S(N)(=O)=O)cn1 N1(C(=O)NC(c2scc(C)n2)(C)C)C(C)CCCC1C c1(OC)sc(C(=O)NC(C)CCNC(c2cnc(S)nc2)=O)cc1Br C1(C)(NC(c2cc(C)c(C)s2)=O)CCCN(C(C2CCC2C)=O)C1 O=C1NCc2cccc(C(N3CCC4(C3)CN(C(=O)C=C3CCC3)CCO4)=O)c21 c1(C(=O)NC2CCC(CNC(C3CC(F)(F)C3)=O)CC2)cc(F)c(F)c(F)c1F CC(C)C(F)(F)CC(=O)NCCC(C)N(C)C(c1ccn(C(C)(C)C)n1)=O Cc1cc(NCC2CC2C2CC2)ncc1S(=O)(=O)N1CC(C)C(C)C1 C(C)(CNC(=O)C=CC1COC(C)(C)O1)(CC(C)C)NC(Cn1c(C)ccn1)=O C12(OC)CC(C(=O)OCc3cccc(-n4nc(C)nc4C)c3)C(C1)C2 C1(NC(=O)C(C2CCOCC2)C)CN(C(c2cc(OC)ns2)=O)CCC1CO C(=O)(CCC[N+](=O)[O-])NCC(C(C)(C)C)NC(C(C(C)C)NC(=O)OC)=O C(=O)(CCCC(C)O)NCC1C(NC(c2c(COC)ccs2)=O)CCC1 N1(C(CN(S(CC)(=O)=O)C)=O)CC(NC(=O)C=CCOC)CC2(CC2)C1 c1(CNC(c2ccncc2-c2cncnc2)=O)ccc(F)cc1Cl C1(CNC(C2CCC(C)C2)=O)CN(c2cc(Cl)ncn2)CCC12CCOCC2 N1(C(c2cc(COC)[nH]n2)=O)CCCC(O)(C(N)=O)C1.C12CCOC(C1)C(=O)N2 c1(C(=O)NCCOC2CCN(C(CC3CC(C)C3)=O)C2)cc(C)c2[nH]cnc2c1 c1(C(=O)NC(C2CSC2)C)cc(CNC(C2CC2[N+](=O)[O-])=O)no1 N1(C(c2cnn(CC)c2C)=O)C2CCC1C(F)C(NC(=O)CC1CNC(=O)O1)C2 CC(C)(C(=O)NC1CC(C)(NC(=O)CNC(c2ccsc2)=O)C1)C1CC1 c1(NC)ccc(C(N2CCC(NC(C3(Br)CC3)=O)CC2C)=O)cc1F N1(C(C(CC=C)OC)=O)CCC(C)(CNC(c2cn(C)nc2C)=O)CC1 c1(C(N(CC(=O)O)CC=C)=O)ccc(C2OCC2(C)C)cc1 C1(O)(CNC(C2CNC(=O)N2)=O)CCN(C(C2CCCCS2)=O)C1 C1(C(=O)OCC)(C(=O)NC2CCCC(NC(C3CN(C(N)=O)C3)=O)C2)CCCCO1 C1(CCNC(c2ccn(CCNC(c3n(CC)ccn3)=O)c2)=O)COC(C)(C)C1 Cc1cccc(Br)c1CC(=O)N(CCCNC(C1CC2CCCC2C1)=O)C c1(C(=O)NCC2C(CNC(C3CC(=O)NC3)=O)C2)cccc(F)c1 N1(C(c2c(CC)con2)=O)CC(CC(=O)N(CC(C)C#N)C)CC1(C)C C(=O)(C(C(C)N(C)C)NC)N1CC(CNC(c2cc(C#N)cs2)=O)C1 c1(C(=O)NCCCN(C(C2C(=C)C2)=O)C(C)C)cnn(CCC(C)C)c1C c1(C(=O)NCC2C(C(N(CCCCC)CC(N)=O)=O)C2(C)C)nnc(S)n1C C1(CC=C)(NC(=O)Cc2n[nH]cc2Br)CCN(C(=O)CS(=O)(=O)N(C)C)C1 C1(C(N2CC(c3cn(CC(O)C(F)(F)F)nn3)C2)=O)C2CCCC(=O)C12 c1(SCC)ccccc1OCC(=O)NCCC(C)N(C1CC1)C(C1CCC1)=O N1(C(C=C(C)C)=O)CCCN(C(=O)C(C)n2cnnn2)C(c2ccccc2)C1 N1(C(CNC(c2n[nH]cc2Cl)=O)=O)CCN(C2CN(Cc3ccc(Cl)cc3)C2)CC1 C(C1CC1)(C1CC1)=CC(=O)NC(C(=O)NCCN(CCOC)C)C1CCC1 C1(CNC(C2C3CC4C(C3)C24)=O)CCCC(CNC(c2csc(F)c2)=O)C1 c1(C(=O)NCC2C(C(=O)NCc3cn(CC)nc3)CCO2)c[nH]c(C#N)c1 N1(C(=O)OC(C)(C)C)CCS(=O)(=O)C(NCc2noc3ncccc23)C1 Cc1cc(O)ccc1C(=O)NCC1(C)CCCN1C(=O)CN1CCC(C)C1 CCCCCCC(CC)C(=O)N1CC2CC(NC(C3CCC=CO3)=O)CC2C1 C1(O)(C(N2CC(C(C)NC(C3CC3Cc3ccccc3)=O)C2)=O)CN(C(N)=O)C1 c1(C(N(C(CCNC(C2(CCC)CC2)=O)C)C)=O)ccc(C(C)C)cn1 N1(C(C(=O)NCC(C)NC(C2C(C(C)=O)C2(C)C)=O)C)C(=O)CCC1=O C(=O)(C(O)CCCNC(C1CC(O)CN1C)=O)N(C)CC1CCC(C)CC1 c1(CC)ccnc(C(N2CCCC2CCC(=O)N2CC(SC(F)F)C2)=O)c1 c1(C(C)C)nc(Br)ccc1C(=O)OCc1csc(Sc2cnc(C(F)(F)F)nc2)n1 C1(C(N2CC(COC)C2(C)C)=O)CCC2CCC1N2C(c1cc(F)cnc1O)=O N1(C(C(C)=C(CC)C)=O)CCC(C(=O)NCC2(C)CC3(CCC3)C2)C1(C)C c1(OCCCC)ccc(C(N2CCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc1 c1(OCC)ccc(NC(N(C)CC2(C)CCN(Cc3nccc(C)n3)C2)=O)cc1 C1(C(=O)NC)CN(C(C2CC2C(=O)NN2CCN(C)CC2)=O)CCO1 c1(C(N2CC3C(CNC(CCCCC)=O)C3C2)=O)c(C)c(O)nc2ccccc12 CC1CCCCC1(CNC(=O)Cn1ncc(C#N)c1N)NC(=O)C1=CCOC1 C1(N(C(=O)C=C2CCC2)CCC)CCN(C(=O)CC2CCCOC2)CC1 Cc1cc(C(=O)N(C(C)CNC(C2CN3CCC2CC3)=O)C)cc(F)c1 N1(C(C(C)CC2CCC2)=O)CCOC(CCNC(C2(C(N)=O)CC2)=O)C1 c1(C(=O)NC2CCCC(CNC(C3CCCOCC3)=O)C2)cccc2occc12 C1(NC(C)=O)CCC(C(N2CCCC2CNCc2nc[nH]c2C(F)(F)F)=O)CC1 c1(C(=O)NC(CC=C)CNC(C2COC(=O)N2)=O)cccc([N+](=O)[O-])c1Cl c1(OC)cccc(C(=O)NCC(C)NC(=O)Cc2cn(C)nn2)c1C c1(C(=O)NC2CCN(C(CC3CCC(C)O3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl C(=O)(CC(C(C)OC)NC(=O)C(CN(C)C)C(C)C)NC(C1CCOCC1)C#C CC(C(=O)N(C)CC1(NC(C2CCC3(CC3)C2)=O)CC1)S(C)(=O)=O C1(NC(C=CC)=O)CN(C(c2ccc(C)cc2OCC)=O)CC2CC12 C(=O)(C(CC(C)(C)C)NC(=O)CC1(N(C)C)CC1)N1CCCC(COC)C1 c1(C(=O)NCCNC(c2onc(C(C)(C)C)n2)=O)occ2c1CCOC2 c1(C(N(CCC)CCNC(C23CC(C2)C(C)O3)=O)=O)cnc2ccc(C)cc2c1 N1(c2nc(SC)nc(C(F)F)c2)C2CCC1CC(NC(C1CC(=O)N(C)C1)=O)C2 c1(C(=O)NCC(CNC(c2ccc(C#N)cn2)=O)F)c[nH]c2cccc(Cl)c12 N1CCOC(CC(=O)NC2CC(C)(O)C2)C1.C12(C(C)(C)C)CC(CC(=O)N)(C1)C2 c1(C(=O)NCC(CNC(C2(C(C)(C)C)CCCC2)=O)O)csc2cccnc12 C1(C(N)=O)CCC(NC(c2c[nH]c(C(=O)NCC3(CCO)CC3)c2)=O)CC1 CCCC(O)C(=O)N1CCC(OCCNC(C23CC(F)(C2)C3)=O)C1 N1(CCCCCNC(c2nc(CCC)sc2)=O)CCN(C(=O)C(C)=C(C)C)CC1 CC(C)CC(CNC(=O)CC1CC=CCC1)C(=O)NCCOCC(F)(F)F Cn1nc(C(=O)NCC2CCN(C(c3sccc3C(F)F)=O)C2)cc1CO N(C(=NCc1ncccc1OC)NC(C)C)C(COC)C(F)F C1(C)(CC(=O)NC2CCC(NC(Cc3cnc(C)s3)=O)C2)CCCCC1 C12(C(=O)NC3C(CC)CC3)CC(C)(CN)C(C1)C2 C1(NC(=O)NCC2(N3CCOCC3)CCN(C)CC2)CCN2CCCCC12 CC(F)(F)CCCC(=O)NC(C)(CNC(c1ccccc1[N+](=O)[O-])=O)C1CCC1 N1(C(c2cc(OC)no2)=O)CC2(CC2)CC1C(=O)NCC1(C2CC2)CCCO1 C12=NC(=N)NC(=NCCN(C)C1=O)N2.c1(OC)cc(CSC)ccc1[N+](=O)[O-] C1(CNC(c2n(CC)nnc2)=O)CCCC2CN(C(=O)Cn3ccnn3)CC12 C1(NC(C(CCC)(C)CC)=O)CC2CCC1CN(C(C13CC(O)C1C3)=O)C2 C1(C(=O)NCC(C)(C)NC(c2c(Cl)ccc(O)c2Cl)=O)COCC2(CCC2)O1 CC1(C)C(NC(=O)C=Cc2cnccn2)CC1C(=O)NC1C(=O)OCC1CO c1(-n2cc(C(C)(C)NC(C3(F)CCOC3)=O)nn2)ccc(C(C)(C)C)cc1 C1(OC)CCN(C(C2CC23CCN(C(=O)CC2CSCCO2)C3)=O)C1(C)C c1(CC)cc(C(=O)NCC#CCNC(=O)C(c2ccccc2)C)ccc1C c1(C(N2CC3C(CCNC(CCSCC)=O)(CC3)C2)=O)c(C)ccc(C)c1O Cc1ccc2sc(C(=O)NCCC(C)(C)NC(=O)C(C)C(C)O)c(C)c2c1 c1(C(=O)NC2C(NC(C=Cc3cnc(C)s3)=O)CCC2)cc2cc(Cl)ccc2o1 Cc1ccn(CC(N2CCC(CN(C)C(c3cn(C4CC4)cn3)=O)C2)=O)n1 C(=O)(CCCCCCCO)N1CCN(C(c2c(C)csc2)=O)C2C1C2 c1(C(=O)NC2C(C(=O)NCC)C2)nccc2c(S(N)(=O)=O)cccc12 c1(NC(C(C)NC(C(C(C)C)(C)O)=O)C(C)C)nc(Cl)nc2c1nnn2C CC(C)C(C)C(C)CC(=O)NCC1(CCNC(C2SCCS2)=O)CC1 C1(C)(CC)CN(C(C2CNC(=O)CN2C(=O)CC2CC(OC3CC3)C2)=O)CCO1 N1(C(=O)OC(C)(C)C)CC(C(=O)NCCn2cc(F)ccc2=O)CCC12COC2 Cc1ncc(C(=O)NCC(C)CN(C(=O)Cn2nccc2C)C)cc1N C1(C(N2CCC(OC)C2C)=O)CCC(O)CN1C(C1C2CCC(C2)C1C)=O C1(O)(CC(=O)N(CCC(C)(C)NC(CN2C(C)CCC2)=O)C)CCOCC1 Cc1cc(C(N2CCC(C)C2)=O)ccc1Br.c12cn(C)c(n1)CNC(=O)N2 Cc1ccccc1-n1nnnc1CC(C)(C)NC(C1CC(N2CC(F)C2)C1)=O C1(C2CC2)(C(=O)NCCN2C(=O)CNC2=O)CN(C(=O)C=C2CCC2)C1 c1(CN2C(C(N3CC4CC3CO4)=O)CC2)cc2ccccc2cn1 Cc1cc(CCC(=O)NCC(C)CNC(=O)CC2COCCO2)cc(C)c1 C(C(=O)NCC1(OC)CN(C(=O)C(O)C(F)F)C1)(C(C)C)SCC N1(CC)CC(NC(C2CSCN2C(=O)C(O)CC2CCCC2)=O)CC1=O c1(C(=O)NCC(C2CCC2)NC(C2CC2C(F)(F)F)=O)ncsc1C1CC1 C1(O)(CC(=O)NC2C(CNC(CCc3n(CCOC)ccn3)=O)C2)CCOCC1 C12(NC(C3(O)CCC3)=O)CCC(CC1)N(C(=O)COC(F)(F)F)C2 C1(CNC(C2=NOC(C)C2)=O)C2CCCC1N(C(C1CCSC1)=O)C2 c1(NC(=O)NCCS(CC)(=O)=O)ccc2c(c1)c(C)nn2C C1(C(=O)NCCN(C)C(c2cnn(CCN3CCCC3)n2)=O)(CC)CC=CC1 N1(C(C2(CNC(c3ccc(CO)o3)=O)CC2)=O)CCN(Cc2n(C)ccn2)CC1 c1(C(N(CCCNC(C2C(C)(CC)C2)=O)C)=O)cnc2sccc2c1 C1(CNC(C(N2C(CC)CCC2)=O)=O)C2CN(C(=O)CP(C)(C)=O)CC12 C1(C(=O)NCC(C)C(=O)N2CC(N3CCOC3=O)C2)Cc2nccn2C1 c1(C(N2CCC(c3nc(C)no3)C2)C(=O)NCCCC)nnc(C2CC2)s1 CC(C)CC(C)CC(=O)NC1CCCN(C(c2cc3ccsc3n2C)=O)C1 C=CC(C)(O)CC(=O)NC1CCC(C(=O)NC2Cc3nccn3C2)CC1 N1(C(c2c(C)n[nH]c2C)=O)CCC2CN(C(=O)C(C)(C)CNC(N)=O)CCC2C1 C1(NC(C2CC3CCC2O3)=O)CCCCN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCCC(COC)OC)(COC)CN(C(=O)C(N2CCCCC2)C)C1 c1(COC)cccc(NC2(CN3CCN(C)CC3)CCC2)n1 c1(C(C2CCCN2C(=O)NC2CN(C)C(=O)C2)O)cc2ncccc2o1 C12(CNC(Cn3c(C(F)F)cc(C)n3)=O)CCC1CCN2C(c1ncoc1C)=O C1(CCC)(NC(=O)CCc2cscn2)CCCN(C(C2CC(F)(CSC)C2)=O)C1 Cc1nc2c(s1)CCCC2C(=O)NC(CC(C)C)C(=O)NO c1(C(=O)NC2C(CNC(=O)C=CC=C(Cl)Cl)CCC2)cncc(Cl)c1Cl CC1CCN(N2CCC(C)C2)CC1.C1(C)(C=O)COCCO1.c12cn(nn1)C2 C(=O)(CCCC(=O)N1CC(CC(F)C(N2CCCC(C(C)(C)C)CC2)=O)C1)OC C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCN(C(C(C)c2cccs2)=O)CC1 c1(C(C)C)ncc(C(N2CCC(N(C(=O)CC3CC4(CC4)CO3)C)C2)=O)n1C c1(NC(N2CC(SCC)OCC2)=O)cc(OC)cnc1F.C(C)(C)(C)OC(N(C)C)=O C=CC(C(=O)NC(c1ccccc1)C(=O)NCCC1COCC1O)OC C1(C(=O)N(CCN(C(CCC#C)=O)CCOCCO)CC)COc2cc(O)ccc2C1 Cc1nc(C)c(C(=O)NC2CCN(C(=O)CNS(C)(=O)=O)C(C3CC3)C2)nc1C c1(NCC(c2ccc(F)cc2F)OCC)ccc(S(=O)(=O)NCCSC)cc1F C1(CNC(CCN(C(COC2(C)CCCC2)=O)CC2CC2)=O)CC(O)CCO1 n1(CC(=O)N(CC(N2CCCC(C)C2)C)C2CC2)nc(C2CC2)n(C)c1=O C1(C2CCCN(C(c3cnn(CCO)c3)=O)C2)(NC(C2(C(C)C)COC2)=O)CC1 C#CCC(O)C(=O)NC12CC(C1)N(C(c1cc(Br)c(OC)s1)=O)C2 c1(C(C2CC2)NC(=O)NC(c2cccs2)C)cccc(O)c1 N1(C(C(C(C)(C)C)NC(c2cc[n+]([O-])cc2)=O)=O)CCC(O)C(F)(F)C1 c1(N2C(C)CC(NC(CCS(=O)(=O)NC)=O)C2)ccc2cnccc2c1[N+](=O)[O-] c1(C(=O)NCCC(C(C)C)NC(=O)Cc2nccs2)ccc(N=[N+]=[N-])cc1 C1(NC(c2c(CC)noc2C)=O)CC2CC1N(C(C13CC1COC3(C)C)=O)C2 CP(C)(=O)CN1CCCC(C(N2CCC(CNC(c3coc(Cl)c3)=O)C2)=O)C1 C1(NC(c2cnn(CC)n2)=O)CC2CCCN(C1)N2C(=O)COC1(C)CCCC1 CC1(NC(=O)Cc2cncnc2)CCCCC1C(N1CCSCC1)=O O=C1CC(C2CC2)(C(=O)NCCC(=O)NCCCC2CCCCO2)C1 c1(C(CNC(=O)C(F)F)N(C(CN(C2CC(C#N)C2)C)=O)C)ccccc1 c1(C(N2CCCN(C(C3CC4(C3)CC4(F)F)=O)CC2)=O)cnn2c1CCCC2 C1(CN(C(c2ccsc2)=O)C2CC2)CCN(C(C2(c3ccccc3)CCOC2)=O)C1 C12(C(N3C(CNC(c4cccc(OCC)c4)=O)CC(C)C3)=O)CCC(C1)OC2C C(CCCC(=O)NCCCCCN(C(=O)C(c1ccccc1)C)C)NC(C)=O N1(C(C2CC(CN(C)C)C2)=O)CC(NC(=O)C(C)Sc2nnnn2C2CC2)CC1 c1(C(=O)NC(CNC(=O)COCCF)(C)C2CC2)cccn2ccnc12 C1(N(CC(C)(C)C)OCCN(CC(C(C(C)OCC2CC2)=O)=O)C)CCCCC1 c1(C(=O)NC2C3CCN(C(C(C)Oc4cccc(C)c4)=O)C32)cc(C)c(C)cn1 N(C1CCNC(=O)c2[nH]ccc21)C(c1c(C)cn(CC)n1)c1nnnn1C C=CCC(C(=O)NC(C(=O)N1CC(OCCOC)C1)C1CCC1)OC C1(CC)CN(C(c2nnc(Cc3ccccc3)s2)=O)CC(C)S1(=O)=O Cc1nc2ccccc2cc1C=CC(=O)N(C)CCNC(C1CC1C(C)(C)O)=O c1(Cc2nn(CCOC(C)=O)c(-c3cc[n+]([O-])cc3)n2)ccc(C(C)(C)C)cc1 C1(CC)CCCC(N=c2cccc(S(=O)(=O)N3CCC(CSC)CC3)[nH]2)C1 c1(NC(C)=O)ccc(CC(=O)C(=O)NCCOCCNC(=O)CCC(N)=O)cc1 CC1(C)CC(C)(C(N2CCC(C3CCCN3C(=O)CCc3cnoc3)C2)=O)C1 CCCC(C)C(=O)N1CC(O)CC1CC(=O)Nc1cn(C)nc1C(N)=O c1(C(=O)NC(C2CCN(C(C3CC(C)(C)CCO3)=O)C2)C)ccc2c(c1)CCO2 c1(C(=O)NC(CCC)C)cc2cccnn2c1 c1(CC)oc(C)cc1C(=O)NCC(C)(C)OCC(=O)NCC1CC(C)(C)C1 N1(C(C2C(CC)C2)=O)CCCC(CNc2cc(C(N)=O)ncn2)C1 c1(CC(=O)N(CCNC(C23CCCN(CC2)C3)=O)CC)ccc2c(c1)CCC2 C1(C(=O)NC(C2CCC2)C)(NC(c2cn(CC=C)nn2)=O)CCN(C)C1 c1(C(=O)NC(CN(C(c2sc(OC)nc2C)=O)CC)C)ccc(C)c(Cl)c1 CCC(C(=O)N(CC(=O)NCC(C)(C)CNC(N)=O)CC)OC.CC(C)C C1(NC(CC2(C#N)CC2)=O)CN(C(c2cc(C3CC3)cc(F)c2)=O)CC1C1CC1 CC1CN(C(=O)C(C)n2cccn2)CCN1C(=O)CCC1CCC(=O)N1 CCCCC(C)C(=O)N1CCCN(C(c2cc(O)cc(F)c2)=O)CC1 N1(C(c2c(C)nc(CCC)o2)=O)CCCC(NC(=O)CCCC(C)C)C1C C1(C(N(CCCCNC(CCC=CC)=O)C)=O)CCCCN1C(C)C C1(N(C)CC2CCN(C(C(C)Cc3cnc[nH]3)=O)C2)CC2CCC1O2 N1(C(=O)CC2CCC3CC3C2)CCN(C(c2noc3c2CCCC3)=O)C2(CC2)C1 N1(C(c2ccnn2C2CCOCC2)=O)CCC(C(=O)N(C2CCC2)C2CC2)CC1 N1(C(C(c2ccc(F)cc2)OC)=O)CCC(O)C(NC(=O)C2=CCOCC2)C1 C1(O)(C(=O)NCC2CN(C(C3ON=C(C)C3)=O)C2)CC2CCC1C2 C1(O)(CCNC(C=CC(=O)OCCCC)=O)CCN(C(c2c(C)cnn2C)=O)C1 C(=O)(C(C)(C)CNC(=O)C(Cn1ccnn1)NC(=O)C=Cc1nccs1)OC C1(NC(c2ccc(C)cc2)=O)(CO)CCN(C(=O)CCCC2CCCO2)CC1 c1(NC(C2CCN2c2ccnc(-c3ccc(Cl)s3)n2)=O)cccc2nc[nH]c12 CCC(C)C(CC(=O)N1CCC(N2CCCC2)C1)NC(=O)CN1CCOCC1 Cc1nc(Cl)ccc1CC(=O)NCC1CC1NC(=O)CC1CCCOC1 n1(C2(C(N3CC4C(NC(C(C(C)C)F)=O)C4C3)=O)CC2)cnc2ccccc12 c1(C(N(C(C)CNC(C2CCC=CCCC2)=O)C)=O)cc2c(nc1N)CCC2 C1(C(=O)NCCC(C)N(C(=O)C(=O)NC2CC2)C)CNC(=O)C(C)(C)C1 c1(C(=O)NCCC(C)(C)NC(c2ccc(OC)s2)=O)cnc2c(n1)CCCC2 c1(OC)cc(CNC2CN(C(c3cn(C)nc3C(F)F)=O)CC2C)ccc1F C(=O)(C1=CC(C)(CCl)C1)NCCOC.C(=O)(C(C)(C)ONC(=O)C1CC1N)OC N1(C(c2cc(C(N)=O)ncc2)=O)CCC2(CC1)CN(C(C13CCC1C3)=O)CCO2 c1(C(=O)NC2CCC(CNC(c3cccc(C)c3O)=O)C2)cc2n(n1)CC(O)CO2 C#CCC(C)(C)C(=O)NCC1CN(C(c2cn(C)nc2C2CCCO2)=O)CC1O c1(C(N2CCC(NC(c3nnnn3C3CCOCC3)C3CC3)C2)=O)scnc1Br N1(CCC)CC(C(=O)NCCCN(C(=O)Cc2cc[nH]n2)CC)CC1=O n1(CCC(=O)N(C(C)C)CCN(C(=O)C(C)(C)C)C)c(=O)oc2ccccc12 c1(-c2cn(CCCCCC=C)nn2)cnc(OC)c(OC)c1 C1(NC(Cc2ccc(C)o2)=O)CN(C(=O)C=Cc2cncn2C)CCC1CO N(C(=NCCCNS(C)(=O)=O)N1CCC(O)C1)CC(CC)(F)F CC1CCCCC1(CNC(c1csnc1-c1ccccc1)=O)NC(=O)CC(F)F C(CCC)(C(O)C(=O)N1CCSC2(CCC2)C1)NC(CCSCCC)=O C(=O)(CS(=O)(=O)CC)N1CC2C(Cn3cc(CCNC(C=CSC)=O)nn3)C2C1 C1(NC(CC(C)(C)O)=O)CC2CCC1CN(C(c1cc3cccnc3[nH]1)=O)C2 CC1(NC(=O)C=C2CC2)CC(NC(=O)C(F)(F)c2cscn2)C1 c12ccc(cc1C)-c1cc(F)ccc1NC2.CCCOCCN(C)C Cc1cn(C)cc1C(=O)NC(C1CC1C(=O)NC(c1nc[nH]n1)CO)C C1(C(C)C)CCCN1C(=O)C(CC1CC1)NC(=O)CC1COCCO1 N1(C(C(F)=CC)=O)CCC2(CC1)CC(NC(c1cnn(C3CCC3)n1)=O)CO2 c1(CC)cnc(Cl)[nH]c1=NC1CN(C(c2nccnc2N)=O)CC2(CCCC2)C1 C12(CNC(COCCCC)=O)CCCC1N(C(=O)C(C(C)C)n1ccnc1)CC2 c1(CCNC(=O)NC2CC(C)N(C3CC3)C2)c[nH]c2cc(F)ccc12 c1(C(=O)NC(CCOC)CNC(c2[nH]nnc2C(F)F)=O)cncc(C#N)c1 N1(C(c2cccc(CC)n2)=O)CCC(CC)(NC(=O)COC2CCOCC2)CC1 CC(C)CC(CNC(=O)CCN1CCOC1=O)C(=O)NC1CCOC12CCCC2 C(N=c1[nH]c(NCc2cccc(Cl)c2)nc(=N)[nH]1)C1C(C)(CO)CCCC1 N1(CCNC(=O)C(=O)NC2CC(F)(F)C23CCC3)CCc2ccccc2C1 Cc1nc2c([nH]1)CC(C(=O)N(CCCNC(c1nncs1)=O)CCO)CC2 N1(C(CCC=C)=O)CCC(C)CC1C(=O)NOCC(=C)Cl c1(CCC)cc(-c2csc(C3CCCCCC3)n2)c(C)[nH]1 c1(C(N2C(CNC(c3c(CC)ocn3)=O)CC(O)C2)=O)nc(Br)n2ccccc12 c1(CNC(CCOCCC)=O)cc(C(=O)NC2CC(F)(COC)C2)ccn1 N1(C(c2c(C)nc(N)cn2)=O)CC2CC(NC(c3cc(C4CC4)cs3)=O)C(C2)C1 c1(C(=O)NC2CC(CCNC(C3C(OC)CCC3)=O)C2)[nH]c(C)nc1C C(CCC(=O)NCCc1cn(CC2CNC(=O)C2)nn1)N(C)C C1(C(N(C2CCN(C(=O)C=Cc3cn(C)cn3)C2)C)=O)CC(F)(F)CCC1(C)C CCCCCCNC(=O)C(Cn1cccn1)C(=O)CN N1(C(=O)NC(C(c2ccc(Br)cc2)OC)C)CCSCC12CC2 C1(NC(CC(=O)NCC)=O)C2CCCN(CCN3CCCCC3C)C2C1(C)C c1(C(=O)NC(C(=O)NC(C#C)(C)C)C2(O)CCC2)cc(Cl)ns1 Cc1ccc(C=CC(=O)NCCNC(C2CC23CCCOC3)=O)cc1C C1(C(=O)NCc2cn(CCC)nc2)CCN(C(=O)CCC(F)(F)F)CC1O C(CC(C)C)(C(=O)NCC1CN(C(C2CS(=O)C2)=O)C(C)(C)C1)OC Cc1ccc(CCC(N2CCCC2C(C)NC(c2nccn2C)=O)=O)cc1 C(CCC(=O)NC1CC(F)(CNC(C2(C(C)(C)C)CCCC2)=O)C1)SC N1(C(C2CCCN(CC)C2)=O)CC2OCCN(C(c3cc[n+]([O-])cc3)=O)C2C1 c1(CCCC)nc(-c2cccc(Cl)c2)nn1C1CCc2ccccc21 N1(C(=O)NC(c2ccccc2)S(C)(=O)=O)CCCC(C2CCCC2)C1 C(=O)(C(O)C(F)(F)F)NCCn1cc(CNC(c2[nH]c(=N)sc2)=O)nn1 c1(C(N(C2CCN(C(C(C(CC)O)(F)F)=O)C2)CC)=O)cncc2nc(O)[nH]c12 N1(C(c2cc(OC)no2)=O)CC(C)(C)CC1CNC(=O)COCc1cc(C)[nH]n1 N1(C(c2c(C)nc(C)[nH]2)=O)CCCCC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)C1 C(CCC(C)C)(C(=O)NCC1CC1CC(C)C)OC.C12(CCCC1)C(=O)N2C c1(NC2CCC(C(=O)OC)C2)cccc(S(=O)(=O)C2CCCC2)c1 C=C(C)C(CC(=O)N(C(C)CCNC(=O)CSc1nc[nH]n1)C)OCC C=CCC(COC)NC(=O)CC1CCN1C(=O)COCC(F)F c1(CN2CC(CC)C2)ccc(Cl)nc1F.n1(CC(=O)N)cc(-c2cncnc2)nn1 N1(C(c2cncc(OC)n2)=O)CC2CCN(Cc3ccc(C(C)(C)C)cc3)C2C1 c1(CC(C)NC(=O)C(C)NC(=O)CCc2nccs2)ccco1 c1(OC)ccc(NC(=O)C(CCO)NS(=O)(=O)C(C)C)c(OC)c1 c1(CC)ccc(O)c(NC(=O)C(C2(O)CCC2)NC(=O)C(C)C2(O)CCC2)c1 N1(C(CC2C(C)(C)C2(C)C)=O)CCN(C(c2ccsn2)=O)CC1C1CC1 C1(NC(c2cc(C)nn2C)=O)CC(C(=O)NCC(O)CN(C)C)C12CCC2 N1(C(C2=CCN(C)C2)=O)CCC2CCC(NC(=O)CCCc3ccccn3)C1C2 N1(C(C2N(C(N)=O)CCC2)=O)CCc2sc(CNC(C3COC(=O)O3)=O)nc2C1 c1(C(=O)OCCCOCCOCC)csc(C(=O)NC)n1 c1(CNC(CNC(c2cc(OC)ncn2)=O)(C)C)ncc(C(F)(F)F)cc1Cl C1(CNC(Cc2c(C)noc2)=O)CN(C(=O)CCC(N)=O)CC1O C1(=O)CC(C)(O)CN1.CCC(C)(CNC(=O)C(=O)N(C)C)OC c1(CNC(CN(C(c2ccnnc2)=O)CC)=O)conc1C N1(C(CCN(C(C)C)C(c2ccsc2Cl)=O)=O)CCOCC(C)(F)C1 Cc1c(C(=O)NCC(CO)NC(=O)C(O)Cn2cncn2)cnn1C(C)C N1(C(Cn2ccc(C(=O)OC)n2)=O)CCCC(N(C)C(C2CCCCO2)=O)C1 c1(CC(=O)NCC(C2(O)CCN(C(CC=C=C)=O)C2)C)ccc2c(c1)CCOC2 O(NC(=O)CC(C)NC(C)=O)CC(=C)Cl CCS(=O)(=O)CC(=O)N1CCC(CNC(C2CCCC2OC)=O)(OC)CC1 CC1CN(C(=O)NC2CNCC3(CCC3)O2)c2c1ccc(Br)c2Cl c1(OCC)nc(Cl)ccc1C(N1CCC(O)(CNC(c2cnncc2C)=O)C1)=O N1(C(C(C)=O)=O)CCN(C(CNC(=O)CCCCF)C(F)(F)F)CC1 CC1(C)CC(C(=O)N(CCO)CC2(NC(C3C4CCCC34)=O)CCC2)C1 N1(C(C2(C(=O)OCC)CC2)=O)CCC(C#N)(NC(=O)Nc2ccc(CO)o2)C1 c1(-c2ncc(CCNC(=O)NCc3nccnc3Cl)s2)ccccc1F CCCCC(O)C(=O)N1CCC2C(C(N3CCCC3C(C)(C)CO)=O)C2C1 N1(C(C(C=C)(C)C)=O)CCC2CCC(C1)N2C(=O)C(C)=CC C12CC13CCN(CC3)C(=O)NC2.C=C(C)CC(=O)NCC=CCC(=O)OC(C)(C)C N1(C(=O)CC2C=CCC2)CCCCC12CC(NC(=O)CSCC1CCCO1)C2 N1(C(c2c(C)oc(CO)c2)=O)CCCN(C(C2(c3cc[nH]n3)CC2)=O)C(CO)C1 C12(NC(C(C)(C)CCl)=O)CCC(NC(c3cc(F)ncc3Br)=O)(CC1)C2 N1(C(C2N(c3ncnc(C)c3Br)CCCC2)=O)CCCS(=O)(=O)CC1C1CC1 S(=O)(=O)(c1cccc2cncc(Br)c12)COC1(C#C)CCC(C(=O)O)C1 C(CCSC)(C(=O)NC(C1CCOC1)C)NC(Cc1cn(CC)nn1)=O C(=O)(C(C(C)C)NC(c1cnc(NCC)nc1)=O)NC(C=C)C1CCC1 C1(C(=O)NC(Cc2cc(C)on2)C)CCC(CSc2c(C)noc2C)CC1 c1(C(=O)NCCC2CN(C(C3CCC3C(F)F)=O)C2)ccc2c(c1)COCC2 C12(C(=O)NCC(C(=O)N(CC=C)CC3CC3)C)CC1CNC2=O c1(CC)cnccc1C(=O)NC1CC1NC(C1CCCCC1n1cc(Br)cn1)=O C1(CC(=O)NCC=CCC(=O)NCC(c2ccccc2)C)CC2CCC1O2 C(=O)(CCC(C)(C)C#N)NCC(C(=O)N(CC)Cc1cnn(C)c1)(C)CC C1(NC(C(CC=CCC)C)=O)COC2CN(C(c3ccccc3N)=O)CC12 CC(C)(CC(=O)NCC1COCCO1)n1cc(CN2CCCC2)nn1 c1(N2CCCC(=C)C2)nc(C)nc2ccc(OC)cc12.C1(NC)CCNCC1 N1(C(c2cccc(CN(C)C)c2)C(=O)NC2CC2)CCCCCC1C N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCCC(NC(=O)CNC(C)=O)C1 Cc1nc(C(=O)NCC2COC(CNC(=O)CSc3cn[nH]c3)C2)cs1 c1(C(N2C(CN(C(c3c(C)oc(C4CC4)n3)=O)C)CCC2)=O)cccc(F)c1F C(=O)(C(CO)C(C)(C)CCCCN)NCC1(Cc2cn(C)nc2)CCCC1 C(CC(C(=O)NCC1CCN(C(=O)CN(C)C)CC1)NC(N)=O)SC c1(CC2CCN(C(=O)NCC(CC)N(C)C)C2(C)C)ccc(O)cc1F Cc1nccc(C(=O)NC(C)CC(C)NC(C2CC3(C2)CC3F)=O)n1 c1(C(=O)NCC(CC=C)NC(C2CC(=O)NC(=O)N2)=O)cc(Cl)ncc1OC C1(NC(Cc2c(CC)con2)=O)CC=C(C(=O)Nc2csnc2OC)C1 Cc1nc(S)sc1CC(=O)NCC1CC1NC(c1ccccc1C(C)(F)F)=O CCC(C)CC(=O)NCC(N1CCC(NC(=O)CCOc2ccccc2)CC1)C C1(C(N2C(CC)COCC2)=O)C2CC(O)C(C2)N1C(=O)Cc1ccoc1C N1(C(c2cccc(Br)c2O)=O)CCC2(CC1)CC2C(N1CCSCC1)=O N1(CCC#C)CCC(C(=O)NC2(CNC(=O)C#CC(=O)N(C)C)CCOC2)CC1 CCC(C)(Cl)CNC(=O)CC1C(NC(=O)COCCC(C)C)CC1O CN1C(=O)CCC1C(=O)NC(c1ccccc1)C(=O)Nc1ccc(OC(F)F)cc1 c1(C(N(CC(O)CN(C2CC=C(C)CC2)C)C(C)=O)=O)c(C)cccc1Br c1(C(=O)NCC(CC)(C)NC(=O)CSc2nc(C)cc(C)n2)c(C)nn(C)c1Cl C(CCCCC(=O)N1CCC(CNC(C2OCCO2)=O)CC1)N(C)C C1(C(N2CCC(CN(C(CC(C)c3ccco3)=O)C)C2)=O)C2CC3C(C2)C13 Cc1cc(N2CCC(c3cc(N)ncn3)CC2)nc(=NCCC2CCCOC2)[nH]1 CC(C)C(C(=O)N1CCOC(CNC(c2cc(Br)n(C)n2)=O)C1)C(C)C N1(C(CC(CCC)(C)O)=O)CCCC2CN(C(=O)CCOC3CC3)CCC12 c1(OC)cc(C)c2cc(C(N3CCOC(c4ncno4)C3)=O)[nH]c2c1 C1(C(=O)NC(C2(O)CCN(c3cc(-n4ccnc4)ncn3)C2)C)CCCCN1C n1(C(C)C)ccc(C(=O)NCC(C)CNC(C2CCC=CO2)=O)c1 Cc1ccc(C(=O)N(CC(=O)NCc2cnc(C)c(C)c2)C2CCC2)cc1O c1(C(=O)NC2CC3CC(NC(CS(=O)(=O)NC)=O)CC32)ccc2c(c1)OCCN2 C(=O)(CC(C)(C)CC(F)F)NCC(C)N(C(C(CC)(O)c1cccc(Cl)c1)=O)C CC1(C)COCC1C(=O)NC1CC1CNC(=O)C(c1ccccc1Cl)(F)F Cn1c(C(=O)NC2Cc3ccc(Br)cc3C2)cc2c(Br)cccc12 C1(=O)NNC(=O)CN2CCC(C2)O1.CC1OCCC1NC(c1cccnc1)=O C1(C(=O)NCC2C(NC(=O)CN3CCCC3)CCC2)COCCOC1 N1(C(CCC(=O)NC)=O)CC23CCCC2(C1)CN(C(=O)Cc1ncoc1C)C3 Cn1nc(C(=O)NCC2(NC(C3CC3CCN(C)C)=O)CCCCC2)cc1O C(=O)(C#CC(C)(C)CNC(=O)C(C)(O)C1CC1)NCC(COC)C(C)C N1(C(c2scc(CCC)n2)C(=O)N(C2COC2)C2CC2)CCC12CCCC(C)(C)C2 C1(NC(c2cc(C)oc2)=O)CCC(N(C(=O)CCOCCN(C)C)C)CC1 C(=O)(C1=CCCSC1)NC1CCCC(CNC(=O)CCN2CCC2)C1 N1(CC(N2CCC(OC)(CNC(=O)CC(=O)NC3CC3)C2)=O)CC(=O)N(C)C1=O CC1CCCN(C(c2ccc(F)c(O)c2)=O)C1CCNC(=O)CSC(C)(C)C c1(N(C(CCN(CC)CC)=O)CCCOC)cc(C)c([N+](=O)[O-])c(C#N)c1 C1(C(C)C)CC(NC(=O)NC(c2ccccc2N(C)C)=O)CS1(=O)=O C1(NC(c2c(C)scn2)=O)CC(CNC(C2(C)CCC(=O)N2)=O)C(O)C1 c1(CNC(C2C(C)(C)C2)=O)ccc2c(c1)CCC2NC(=O)C#CC1CCCOC1 C1(N(C(=O)CN(C)CCO)CCC)CCN(C(c2cncnc2C)=O)CC1 N1(C(c2cccc(NC(CC=C)=O)c2)=O)CCCC(NC(C)=O)CC1 Cc1nnc(CSC(C)(C)C)s1.N12CC(O)(C1)C1CC(O1)C2=O c1(C(N(CC(CC)Nc2onc(C)c2C)CC)=O)cnc2ccccc2n1 C1(C(=O)OCC)C(C2CC2)CCN1C(c1cc(O)cc(F)c1F)=O Cc1nc(C(=O)NCC2C=CCN2C(c2csc(-c3ccoc3)n2)=O)c(C)s1 C1(NC(C2CCCO2)=O)CC2CCCC2C1.C12(CC13CCC3)C(=O)NC2 CC(=O)C(C)CC(C)C(=O)N1CC(N(C)C(c2ccc([N+](=O)[O-])cc2C)=O)C1 n1(CC(=O)NC2(CC)CCCN(C(=O)COC(F)F)C2)cnc2ccccc12 CC(C)(CC(=O)N1CCCC(NC(C2CC(n3cnnc3)C2)=O)C1)C(F)(F)F CC(C)CC(C)C(=O)N1CCC(C)(CNC(C2(c3ccc(F)cc3)CC2)=O)C1 N1(C(C2C(C#C)C2)=O)CC(OC)C(OC)C1CNC(C1CCC(C(N)=O)C1)=O N1(C(C(CCSC)O)=O)CCC2CCN(C(c3cncnc3C3CC3)=O)C2C1 C(CCC(=O)NC(C)CNC(C1(CCc2ccccc2)CC1)=O)OC C1(NC(c2n(C=C)ncc2)=O)CC2(CCCCN2C(C2CCN(C)C2C)=O)C1 c1(C(N2CC(C3OCCN(C(CC(C)(C)OC)=O)C3)C2)=O)cnc2[nH]c(=N)sc2c1 Cc1cc(N)cnc1C(=O)NCC(C1CC1)NC(=O)Cn1nnc(C(C)(C)C)n1 c1(C(=O)NCC(CC)(CC)NC(c2nccnc2N)=O)ccc(C(C)C)c(N)c1 N1(C(C(C)(O)C2CC2)=O)CCN(CCNC(=O)C=CC2CCC2)CC1 c1(OC(CC)C(=O)NCC(CC(C)C)NC(=O)CNC(C)=O)cccc(Cl)c1 C(=O)(C(C)CC(C)C)Nc1nc(C)c(C(=O)NCC(C)CSc2ccccc2)s1 C=CC(C)CC(=O)NC1(CNC(=O)C(C)(C)C2CCCC2)CC1 C1(C(=O)OC)CN(CC2CCCOC2C(C)(C)C)C(C)(C)CO1 C1(CCC)CN(C(c2cc(C(C)C)n(C)n2)=O)CCN1C(C1CC2CC2C1)=O CCCC(C)C(C(=O)Nc1ccccc1Cl)N1CC2(CC2)C1 c1(NCCC(CNC(=O)CCc2ccc(O)nn2)O)nc2ccc(N)cc2s1 C1(C2CCCOC2)(NC(c2c(CNC(C3CC(CC)OCC3)=O)occ2)=O)CC1 C12CN(CCC1C(F)(F)F)CCN2C.C(C)(C)(C)OC(=O)OCC CCCC(C(=O)NC)NC(=O)CC1CCC(NC(=O)C(F)=CC2CC2)CC1 C1(OC)C=CCN(C(=O)C(Cc2ccco2)NC(c2cnsc2)=O)C1 C1(F)(CNC(CC2C(=O)NC(=O)N2)=O)CCCN(C(C2(C3CCCO3)CC2)=O)C1 c1(C(N2CCCC(NC(c3cc(C)[nH]c3)=O)CCC2)=O)cc2n(n1)CC1(CC1)C2 CC(C)C(C(=O)NC1CCN(C(c2ccnn2CCF)=O)CC1F)C(C)C N1(C(c2c(OC)csc2)=O)CC(NC(=O)CC=Cc2ccccc2)CC(C)C1 c1(C(=O)NC2CC(F)(CNC(CN(C)CCO)=O)C2)ccc(Cl)cc1Cl C(=O)(C(CC(F)(F)F)c1ccc(Cl)cc1)N(C)CCNC(c1cccc(C#N)c1)=O n1(CC(N2C(C(C)NC(=O)CNC=O)CCC2)=O)ncn(C)c1=O C1(NC(C23CC(COC)(OC2)C3)=O)CN(C(=O)CN2CCC(C)CC2)CC1(C)C c1(C(=O)NCC(OC)OC)cc(-c2cnn(CC(C)(C)O)c2)c2cc[nH]c2c1 c1(CC(N2CCCC(NC(C(CC)NC(C)=O)=O)C2)=O)ccc(OC)cc1F N1(C(C(CC)CN(C)C)=O)CCC2(CC2)CC1C(=O)Nc1cnn2c1CCCC2 c1(C(=O)NCCC2CCN(C(C(CCCOC)C)=O)C2)cc2cnccc2[nH]1 N1(C(C2(O)CCN(c3ncc(OC)cn3)C2)=O)CC(C)(C)OCC1(C)C C(CCC(=O)NC1(CNC(c2cnn(-c3cccnc3)c2)=O)CCOC1)N(C)C C1(COC(c2cccc(OC(C)C)n2)=O)CCN(C(=O)C(O)CC(C)C)CC1C c1(C(N2CC(CNC(C(C)SCC)=O)C(C)C2)=O)c(O)nnc2c1CCC2 c1(C(=O)NCCCCC(C)NC(Cn2nnc(C)n2)=O)sc2sccc2c1Cl c1(N(CCCNC(=S)NCc2cccnc2)C)ccc(F)c(Cl)c1F C(=O)(CC(C)(C)CC(F)(F)F)NC(C1(CNC(c2nc(CO)co2)=O)CC1)C C(=O)(C#CC1CCOCC1)NC1CC(NC(c2c(C)ccc(CC)c2)=O)C(O)C1 N1(C(C2(c3cccc(OC)c3)CCCC2)=O)CC(OCC(F)F)CC(O)C1 Cn1cnnc1CCC(=O)NCCC1(C(=O)N(CC(N)=O)CC(N)=O)CCC1 CCC(C)(C(=O)NC)OC.C(=O)(CCC(C)OC)C1(OC(C)C)CN(C(C)=O)C1.C1CCS1 S(=O)(=O)(c1ccsc1C(=O)OC)N(CC(CCC)O)C C12(CNC(C(CCC)C)=O)CCC(CC1)N(C(=O)CC1(CSC)CC1)C2 c1(C(N2CCC(C(CNC(COC)=O)(C)O)CC2)=O)c(C)cccc1[N+](=O)[O-] N1(C)CCC2CN(CC=C(C)C)CC12.c1(SC)cc(C(=O)N(C)C)oc1C N1(C(CSCCCC)=O)CC(CNC(=O)C(C)OC)C2(CCC2)C1 C1(CC)CC(C(=O)NCCCn2ccnn2)CCN1C(=O)C=C(C)C(C)(C)C CC1(C)CC(NC(c2cnsc2)=O)CN1C(=O)CSCC(F)F c1(C2(C(=O)NC3C(CNC(C(C)C#N)=O)CC3)CC2)ccc(Cl)cc1 C1(C(=O)NCC(CNC(C2(CC(=O)OC)CCCC2)=O)OC)CC2(CCC2)CO1 C1(C(C(=O)NC2(CNC(C(COC)O)=O)CC2)C)CCC(C)(C)CC1 Nc1cc2c(cc1C(=O)NC1CCCCCN(C(c3occc3F)=O)C1)CCC2 c12cnc(c(Br)c1)[nH]2.c1(C(N(C)CCOCCO)=O)nccs1 N1(C(c2c(C(C)C)nns2)=O)CCC2(NC(c3csnn3)=O)CCCCC12 C1(NC(c2c(C)oc(C(C)C)c2)=O)CCN(C(=O)COCC(F)F)CC1F C1(O)(C(C)NC(C(C)CN(C)C)=O)CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1 N1(C(C(C(C)C)F)=O)Cc2ccccc2C(NC(c2ccnn2CCN(C)C)=O)C1 c1(CC(=O)NCC(CNC(=O)CCc2nncs2)OC)ccc(F)c(Cl)c1F C(CS(=O)(=O)NCCC(=O)NCC1(O)CN(C2CCC2)C1)OCC.C1(=O)CN1.SCC N1(C(C2C3CN(C(C(C)OCC=C)=O)C2C3)=O)CCCC(N=[N+]=[N-])C1 C1(OCCCC)CCN(C(=O)C(=O)NCC2(CNC)CC2)C1 C(=O)(NNC(=O)CC(C)(C)C1CC1)C(=O)OC(C)(C)C.C(CC(C(N)=O)N)OC c1(-n2ncc(C)c2)cccc(C(=O)NC2CC(CNC(C3CCC(C)O3)=O)C2)c1 N1(c2ncc(CN3C(C)CCCC3C)s2)C(=O)c2ccccc2C1=O N1(C(=O)CN2CC=CC2)CCC2C(CCCN2C(C2(CO)CC2)=O)C1 c1(C(N(CCCOC)C(c2cccs2)=O)=O)cc(CC(C)C)on1 c1(C(N(C2CC2)CC2N(C(CCCCC#C)=O)CCC2)=O)cc2ncccc2s1 CC(C)CC(=O)C(=O)NCC1CCC(N(C)C(C2CCCCC2)=O)CC1 C1(NC(c2ccc(C#N)o2)=O)CCCC(NC(=O)CCc2ccncn2)CC1 Cc1ccc(C=CC(N2CCC(O)(C(C)NC(=O)C(C3CCCCC3)=O)C2)=O)o1 N1(C(=O)CC2CC(C3CC3)C2)CCC2CCCC12C(=O)NCC(C1CC1)C1CC1 c1(C(=O)NCCCC(C)NC(C2COCCOC2)=O)ccccc1C(F)F c1(OCC)cc(Cl)ccc1C(N1CC(NC(=O)C(C)(C)C(C)O)C(C)(C)C1)=O CC1C2CCC(C2)C1C(=O)NC(c1ccccc1)COc1cccc(Cl)c1 N1(CCOCC#C)CCN(C(=O)NCCc2ccccc2C#N)CC1C C(=O)(CCCC(CC)CC)NC1CCN(C(COCC)=O)CC1 C1(C(=O)NC(CCCC)COC)CN(C)CCN1C(c1cc([N+](=O)[O-])n[nH]1)=O C=CCC(CNC(=O)CN(C1CCSC1)C)NC(=O)Cn1ncc(Br)n1 C1(C(=O)NC(CC)C2CC2)(NC2CC2C(=O)SCCCC)CCC1 C1(NC(c2cc(C(N)=O)ncc2)=O)CS(=O)(=O)CC1NC(=O)CN(CCO)C1CC1 Nc1cnc([N+](=O)[O-])cc1C(N1CCCC(NC(=O)CCS(N)(=O)=O)CC1)=O Cc1cc(=NC(C)c2c(Cl)ccc(F)c2Cl)[nH]c(NCC2C3COCC23)n1 c1(SC)cc(C(N2CC3CC(NC(=O)CCC4CCC4)C2C3)=O)ccc1[N+](=O)[O-] N1(C(c2cc(C)on2)=O)C2CCC1C(C)C(NC(c1ccoc1Br)=O)C2 c1(C(N(C(C(=O)N(CC=C)C(C)C)C)C)=O)cnoc1 N(S(=O)(=O)N1CCCC1C)(C1CCCCC1)CC C(C)(c1ccco1)=CC(=O)NCC(COC)NC(=O)CC1CC1C(C)C CC1=C(C(=O)NC(C)CN(C(=O)C(C)C)C)Cn2nnnc2N1C C#CC12CC(CN1C(=O)CC(C)CNC(=O)C=CC1CCCC1)C2 c1(OC)cc(S(=O)(=O)NC(=O)CC2(C(F)F)CC2)c(Cl)cc1Cl c1(C(=O)NC2C(C)(CNC(C3(OCC)CCC3)=O)CCC2)cc2n(n1)CC(F)C2 C(C)(C(=O)NCC=CC(=O)NC(c1ncc[nH]1)C)NC(C)=O CC1CCN(C(=O)C(=O)NCC(C(C)(C)C)NC(c2nc(Cl)cs2)=O)CC1 C1(C(=O)NC2C(OC)CCC2)CCC(CNC(=O)CCC2(C)CC2(F)F)CC1 C#Cc1ccc(C(N2CCCCC2C(=O)NC2C=CCCC2)=O)cn1 C1(CNC(C(C)OCCCC)=O)CN(C(=O)C=CSC)CC12CCC2 c1(C(N2C3C(CNC(C(C)CN(C)C)=O)C(C3)C2)=O)nc(O)nc(O)c1N C(CCCC(C)(C)C)N(C(=O)NC(C)C)C C1(CNC(C2=C(C)CC2)=O)CC2(CCN(C(c3cnc(C)[nH]3)=O)CC2)CO1 c1(C(=O)NC2CC(NC(C3(C)CCC(C)C3(C)C)=O)C2)cc2c(F)cccc2[nH]1 NC1CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC12CCC2 C(CCCC(CO)NC(C1CCC(F)(F)C1)=O)NC(=O)CNC(C1CCCC1)=O c1(C(=O)NCCC2CN(C(=O)CCN3CCC(O)CC3)C2)cc(O)nc(Cl)c1 c1(SCC2CCN(C(C(c3ccc(SCC)o3)C)=O)C2)ccc(Cl)cc1 c1(C(=O)NC23CCN(C(C4CC5(C4)CC(F)C5)=O)CC2C3)cccc2cncn12 CC(C)C(CCNC(c1coc(Cl)n1)=O)NC(C1(Cl)CC1(C)C)=O CC1=C(C(=O)NCc2cncc(C(N3CCCC3CCN(C)C)=O)c2)CCO1 CCCCCC(C)CC(=O)N1C2CCC1CC(N(C(=O)C(C)(C)OC)C)C2 C(c1ccc(Cl)s1)=CC(=O)N(C1CCCC1)CCNC(C1CN(C(N)=O)C1)=O C1(CC(=O)N(CCN(C(=O)Cc2c(Cl)cnn2C)C)C)CCC(=O)N1C CON1CCC(C(=O)NCCC2CN(C(c3cc4n(n3)CCC4)=O)C2)CC1 C1(CCC)CCc2ccccc2N1CCNC(=O)Nc1cc(C(F)(F)F)ccn1 C#Cc1ccc(C(=O)NC2CC(NC(=O)C(c3ccc(Cl)s3)C)C2)o1 c1(N(C2CCN(C(C3CCN(C)C(=O)C3)=O)CC2)C)ncc(Cl)cc1[N+](=O)[O-] N1(C(C(COC)NC(C)=O)=O)CCCN(C(C2C(F)(F)C23CC3)=O)CC1 c1(C(N(CC(C)C#N)C)=O)cc(CNC(=O)C(C)OCOC)no1 C1(NC(c2c[nH]ccc2=O)=O)CN(C(=O)C(O)Cc2cnc[nH]2)CC12CC2 S(=O)(=O)(c1ccc(C#N)cc1)N1CCC(NC(c2c(C)nn(C)c2Cl)=O)C1 N1(C(c2cc(N3C(C)COCC3)ncc2)C(=O)NCC(F)F)CCOC2(CC2)C1 c1(C(=O)NCC(CC=C)NC(C2C=CC=CC=C2)=O)cc(C)c(N)cc1F C12(NC(CCCC(C)O)=O)CCCN(C(c3c(F)cccc3Cl)=O)CC1C2 C12CCOCCN1C2=O.C1(CC)CC(C)CN(C(=O)COC(C)=O)C1 c1(OC)cc(C)c(C(=O)N(C(C)CCNC(=O)CCc2cccc(C)c2)C)cn1 c1(C(=O)NCC2CC3CC3N2C(c2sccc2F)=O)cc2cc(Cl)ccc2o1 c1(C(=O)NC(C2CN(C(=O)C(C)(C)C(C)O)C2)C)cc(C#N)[nH]c1C C1(C)(COC)CN(C(=O)C(C)CNC(=O)CSc2nc[nH]n2)CCO1 c1(NC(=O)NCC2C(C)CCCC2)nc2c(Cl)c(Cl)ccc2s1 C1(CCNC(=O)CC2CC(F)(F)C2)CCCN(c2nc(C3CCCCC3)ns2)C1 N1(C(Cc2ccn(CC)n2)=O)CCC2(CCCCN(C(=O)C3=CC4CCCC34)C2)C1 C1(C(=O)NC(CCCNC(CSC)=O)C)CCCN1S(=N)(=O)N(C)C C(c1ccc(Cl)cc1)=CC(N1CC(NC(C2(CCC=C)CC2)=O)C(OC)C1)=O C1(NC(c2ccnc(OC)c2F)=O)CCCN(C(=O)CCc2ccon2)CCC1 C1(C(=O)NCCCN(C(=O)Cc2ccc(F)cc2)C(C)C)CC2OC1C1CC21 C1(C(=O)O)(CF)CCN(C(C2CCCC3CC23)=O)C1.c1(C(=O)N)ccc(CO)nc1 C(CC(=O)N(CCC(C)C)C1CC1)O.C(=O)(CS)NCCOC.C1(=O)CN1 N1(C(CC(C)NC(N)=O)=O)CCN(C(C2(n3cncn3)CC2)=O)C2(CCC2)C1 C(CCCCCC(=O)N1CCC(NC(c2cnn(CCF)c2)=O)CC1C)SC N1(C(C)(C)C)CCN(C(=O)C(N2CCC(CN)(CF)C2)=O)CC1 C(=O)(C1CCc2c[nH]nc21)NCC(CNC(c1n[nH]c(C)c1Br)=O)F C(CCCNC(c1cnc(C(C)(C)C)s1)=O)(c1ccccc1)NC(C(C)C)=O C1(OC)COCC1NC(=O)C(CN(c1ccccc1)C)NC(=O)CC#N N1(C(C(C)(C)OC)=O)CCC(O)(C2(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)CC1 C1(NC(C=NOC)=O)CN(C(C2CC(=O)N(C(C)C)C2)=O)CC1n1ccnn1 N1(C(=O)CC2CCCCC23CC3)CCC2(CCCN2C(c2ccc[nH]2)=O)C1 c1(C(C(=O)N2CC(OC(F)F)C2)NC(C(C)NC(CC)(C)C)=O)ncnn1C C(=O)(CC1COCc2ccccc21)NC1CCC(NC(c2c(C)snn2)=O)C1 CC(C)CC(C(=O)N1CC(C)C1C(N1CCSCC1)=O)N(C)C CCC(C)C(C)(O)CNC(=O)CC1(N(C)C(c2cncc(C)c2)=O)CC1 c1(C(N)=O)cc([N+](=O)[O-])ccc1NC(=O)C1CC1.C1(C)C(C2CC2)N1 C1(NC(C(C(C)C)C)=O)C(C)(C)CN(C(c2ccc(C(N)=O)s2)=O)CC1(C)C CC1CC(C(=O)Nc2c(F)cccc2Cl)CC(C)C1 C1(C2CC2)(C(N2CC(CNC(COC(CC)C)=O)C(C)C2)=O)CC=CC1 C1(CN(C(C(C)C2CCCC2)=O)C)CCC(NC(C2(C)CC=CCC2)=O)CC1 c1(OC)cccc2cc(C(=O)NCc3ccnn3C(C)C)oc12 c1(OC)ccnc(F)c1C(=O)NCCC1CC(NC(c2ncoc2C(C)C)=O)C1 CCCC(C)CC(=O)N1CCN(C2CN(C(=O)C(F)C(C)C)C2)CC1 Cc1cc(C)nc(SCC(N2CCN(C(=O)CCC(F)(F)F)C(C(F)F)C2)=O)n1 C1(C(=O)NCCN(C(=O)CN(C)C(=O)N(C)C)C(C)C)C2CCCCCC12 c1(C(=O)NC2C(CNC(C(C(C)(C)C)O)=O)CC2)ccc2nc(O)[nH]c2c1 C12(CNC(c3cc(COC)on3)=O)CCC1CN(C(=O)C(F)(F)c1nccs1)C2 C(=O)(C(C)(F)C(C)(C)F)N1CCCC(N(C(c2ccc(CC)c(Cl)c2)=O)C)CC1 CCC(C)C(C)C(=O)NC1(CO)CCCN(C(C)C(=O)NC(C)C)C1 n1(CC)cc(CNC(=O)C(CC2CC2)NC(C2CCCO2)=O)cn1 CC1CC(CNC(C2(C)CCSCC2)=O)CN(C(=O)CSc2cccs2)C1 O=C1CC(C(=O)NC2CN(C(c3cccnn3)=O)CC2n2ccnn2)CCN1 CCCC(Cc1ccccc1)N(C(c1nccs1)C(=O)NCCC#N)CC(C)C CCCCC(C)(c1nnnn1CC(F)F)NC(CC(C)(C)C)c1ccccc1 CN1CCC(C)(C(N2CCC(C)(CCNC(=O)CC3CCC3)C2)=O)C1 C1(CNC(C)=O)CC(F)(F)CN1C(=O)C(F)OC(F)(F)F.c12ccc(cc1)n2C CCCCC(=O)N1CCCC1CC(C(=O)OC)NC(=O)CC=C(C)C C1(CNC(C(C2CCCC2)NC(c2cn(CC)nn2)=O)=O)OCCC1(C)C c1(C(=O)NCC(C2CC2)NC(CC2ON=C(CC)C2)=O)c[nH]c2c(Cl)cccc12 C1(NC(C=CCN(C)C)=O)CC(CNC(=O)C=CI)C1 C1(N(C(C2CN(CC(=O)OC(C)(C)C)C2)=O)OC)CCC(Sc2ccccn2)CC1 C1(NC(C(COCC)NC(C23CCC(CC2)CO3)=O)=O)CCCOC12CCC2 c1(CNC(C2C(C(=O)Nc3ccc(C)cc3Br)C2)=O)c[nH]nc1S(N)(=O)=O N1(C(C2C(CC)CCO2)=O)CCN(C(c2ccc(C)o2)=O)CC1COC N1(C(c2c(C)cco2)=O)CC2CC(C)N(C(=O)C(C)O)C2C1 c1(OC)cc(CN2CCC(F)(F)C(C(=O)NCc3cn[nH]c3)C2)cc(Cl)c1O C1(CNC(=O)CC(F)(F)F)CC2CCC1N2C(C1(F)CCOCC1)=O c1(C(N2CC(NC(c3c(CC)n(C)nn3)=O)C(C)CC2)=O)cnc2[nH]cnc2c1 c1(C(=O)NC(C2CCCN2C(C2CCCO2)=O)(C)C)nc(CO)n2ccccc12 C(=O)(CC1CCC(C)(C)c2ccccc21)NC(C(C)(C)OC)C(C)C C1(NC(CC(C)C2CC2)=O)CN(C(=O)CCCC2CCCCC2)CCC12CCC2 CCC(C)(F)C(=O)NCCCN(C(=O)C(C)N(CC)CC)C c1(C(=O)NC23C(CN(C(C(C)OC)=O)C2)CCCC3)ccc(N=S(C)(C)=O)cc1 c1(C(=O)NC2(CNC(c3c(C)occ3)=O)CC2)ccc(F)cc1Br Cc1[nH]nc(NC(=O)CN(CCO)CCn2ccnn2)c1C C1(C(=O)NCC(C2CCCC2)NC(C(CCC)NC(C)=O)=O)CC2COCC2C1 c1(NC(C(CCOCC)N)=O)c(C)[nH]c2ccc(Br)cc12 N1(C(C2C(CC)CN(C(=O)C(=CC3CCCC3)C)C2)=O)CCOCC(C)C1 C1(C(N(CC(C)NC(c2c(COC)n(C)nc2)=O)C)=O)CC2OC(C)(C)OC2C1 CCCC(CC)CCC(=O)N1CCCCCC1C(=O)NC1C(C)(C)C1(C)C n1(CC)cnc2nc(N(C)CCSC)nc(N3CC(C)C(C(F)(F)F)C3)c12 c1(NC(COC)CC(C)(C)C(=O)OCC)c(C)nc2c(OC)cccn12 N1(C(C)=O)CCC(CC(=O)N(CC(C)CNC(=O)CSc2n[nH]c(C)n2)C)CC1 c1(NC2C(C(C)(C)C)CCC2)ncc(S(=O)(=O)NC2CCn3ccnc32)cc1Cl C1(C(N2CCCC(C(N3CCCC(C(=O)NC)C3)=O)C2)=O)CCC(C)=C(C)C1 N1(C(c2ccc(OCC#C)cc2)=O)CCC(NC(=O)CCC2CCOC2)C(O)C1 c1(C(N2CC(C(C(=O)NC(CC)(C)C)OC)C2)=O)cc([N+](=O)[O-])n[nH]1 CN1CCC(C(=O)NCC2(C(N)=O)CC2)(NC(C2CC2C(F)F)=O)C1 N1(C(c2nc(C)oc2)=O)CCCC2CC(NC(=O)CC3OCCC3(C)C)CCC12 c1(C(=O)OC(C#C)C(C2CCC2)OC)cccc(OCC)c1 c1(C(N2CCC(N(CCC)C(c3c(C)noc3C)=O)C2)=O)cc(F)c(O)c(F)c1 C12(NC(CC3(OC)CCOCC3)=O)CCC(CC1)N(C(=O)C(C)CS(C)(=O)=O)C2 C(=O)(CCC(C)CC)NCc1c(C(=O)NC(CCCC)CO)n[nH]c1 C(=O)(C(O)C(F)(F)F)N(CC(CC)NC(=O)C(C)(C)c1ccccc1)CC CCC(C(=O)OC)C(=O)NCC(CNC(=O)CC(C)(C)F)CO C1(NC(c2c(CC)noc2)=O)CC2C1CCN2C(=O)COCCOCCO CCCCC(O)CC(=O)NCC1CC2CCC(C1)N2C(=O)C=CC(C)(C)C CC1=C(C(=O)N(C2CCC3CN(C(c4cn(CCOC)nn4)=O)CC23)C)CCCC1 N1(C(c2cnn(C(C)C)c2F)=O)CCC2(CCCN2C(c2cncnc2)=O)C1 Cc1ccc(NC2CCCC(C(=O)OCC(F)(F)F)C2)nc1 C1(NC(C2C(NC(C(C)C#N)=O)C3CCC2C3)=O)CCCN2CCCC12 c1(NC(C(=NOC(CCCC)C(=O)OC)C)=O)ncccc1S(=O)(=O)CC C1(C(F)(F)F)(C(=O)OC)CCCCN1C(C1C(C)(C)C1(C)C)=O C1(CN(C)C(C2(C)CCCO2)=O)CCCN1C(C1(CC2CC2)CCCC1)=O C(C(C)(C)C(=O)NCc1ccc(C#N)s1)N(C(C(SC)SC)=O)C CC(CCCCCO)NC(C1(F)CN(C(C2CCN(C)C2=O)=O)C1)=O c1(C(=O)NCC(CC=C)NC(c2c(CO)noc2C)=O)ccc(N)c([N+](=O)[O-])c1 C1(CC(=O)Nc2cccc(SCCCO)c2)C2CCCC2N1C(=O)C(F)F C1(NC(C2C(C=C)C2)=O)(CO)CCN(C(c2cnc(OC)c(Br)c2)=O)C1 N1(C(C(C)=C(C)C)=O)CCCN(CCNC(C2CCC(O)C2)=O)CC1 N1(C(=O)Cn2ncnn2)CCN(C(C2CC2(Cl)Cl)=O)C2CCC12 Cc1ccc(CS)cc1.C12(CN(C(=O)Cn3nccn3)C1)OCC(=O)N2.C(C)(C)O N1(C(CCN(C(C2CC2C(F)(F)F)=O)CC)=O)CCC(C(=O)OC)C1 C1(C(N(C2CCCNC2=O)C)=O)C2CC3C(C2NC(=O)CCc2cnn(C)c2)C13 C1(C(=O)NCC(=C)CCNC(C2CC(CC(C)(C)C)C2)=O)CCN(C)C(=O)C1 C1(C(=O)NCC(C2CCCCC2)NC(c2nocc2Cl)=O)COCCOC1 C1(=O)CCCCN1.C(=O)(CCC=CC)NCCOCCC=C N1(C(C2N(C(CC(C)C)=O)CCCC2)=O)CC=C(CNC(C2CCCO2)=O)CC1 CC(C)(C)CCCCC(=O)NCC12CC(NC(=O)CCc3ccnc(Cl)c3)(C1)C2 C(=O)(CC(C)(C)CNC(=O)C(C)(C)C(N)=O)N1CCC(C(=O)NC)C1C N1(C(c2c(C)ccnc2O)=O)CC2CCN(C(=O)CC3CC34CC4)CCC2C1 C(C)(C)(C(=O)N1CC(CCNC(c2coc(-c3ccccc3)n2)=O)C1)OCC C1(C(N2CC(F)(C(=O)OC)C2)=O)C(C)CCN1C(=O)C(C(C)OC)N(C)C CCC(CC)C(CNC(N1CCOCC1(C)C)=O)N1CCCC1 N1(C(c2c(CC)n(C)cc2)=O)CC(CNC(=O)CN2CCCNC2=O)CC(C)C1 CCCC(C)CC(=O)NCC1CC(C(F)(F)F)CN1C(C1CC(F)(F)C1)=O CCC1=C(C(=O)NC2CCC2NC(C2CC(C3CCOCC3)=NO2)=O)CCCO1 C1(C(=O)NCc2cccc(CN(C(=O)CCC(F)(F)F)C)c2)CC(=O)NC(=O)N1 c1(CSC)ccc(C(N2CCCC2CNC(=O)C2=CC(C)CC2)=O)cc1[N+](=O)[O-] Cc1ccccc1CCC1CCCN(C(=O)C(=O)N(c2cccc(Cl)c2)CCO)C1 c1(C(N(C2CN(C(C3(CO)CCCO3)=O)C2)C)=O)cccc(-c2cccnc2)c1 C(=O)(C(C)(C)C(O)CC)CC(NC(NC(C=C)C)=NCC1CCCCC1)C.N Cc1c(F)ccc(C(=O)N(C)CC2(NC(=O)C(c3cnn(C)c3)C)CC2)c1Cl N1(C(CNC(CCC)=O)=O)CC2CC(C(N3CC(C)(C#N)C3)=O)C(C2)C1 c1(C(=O)NCC(CNC(C(C=C)c2ccccc2)=O)O)cccc(C(=O)NC)c1 C(=O)(CC(F)(F)C(F)(F)F)N(C1CCN(C(C2CC2(F)F)=O)C1)CC n1(CCCCCC)nc(SCC(N2CC3COC(C3)C2)=O)c2ccccc12 C1(C)(C(N(C)CC2(O)CN(C(C3(SCC)CC3)=O)C2)=O)CCCC1C N1(CCOC)CC2(CN(C(C3CCOCCN3C(=O)COC3CCCC3)=O)C2)C1 CCCCC(O)CC(=O)NC1(CO)CN(C(=O)C=CC2(C)CCOCC2)C1 CC(C)CC(F)C(=O)NCC1CCCCN1C(=O)CCc1ccoc1 C1(C(C)NC(C2(OCC)CCC2)=O)CCCN1C(=O)CC1(C)CC1(F)Cl C(=O)(C(C)(C)CC(F)F)N1CC(C(=O)NCC(F)CO)CC(C)C1 c1(C(C(=O)NC(c2ccc(C(F)(F)F)cc2)CC)(F)F)cc(C)ccn1 C(=O)(C(O)C(C(C)C)OC)N1CCC(C(=O)NCC(C)(COC)CO)(OC)C1 CC1COC2(CCN(C(=O)NC34CCC(C)(CC3)OC4)CC2)C1 N1(C(C(CC)=CC)=O)CCC(NC(c2ccc(N3CCOCC3)nc2)=O)C(F)C1 Cc1nccn2ncc(C(=O)NCCCc3ccc(Cl)cn3)c12 CC1=C(c2ccco2)CN(C(C2C3CC3C3CC23)=O)CC1 N1(C(CC(=C)C)=O)CCCC1(C)CNC(c1cn(C(C)(C)C)cn1)=O C#CCCCCCC(=O)NCC1CCN(C(c2cnn(CCO)c2)=O)C1 c1(C(=O)NCc2cccc(NC(c3cnn(C)c3Cl)=O)c2)cnn2c1CCC2 N#Cc1cccc(S(=O)(=O)N2CCC(O)CC2C(=O)N=c2[nH][nH]cc2C)c1 C1(NS(=O)(=O)CC2CCCC(F)C2)CC2(CCC2)C1 CCC(CC(=O)NC1CC2(CC2)C1)NC(=O)C(O)Cn1cncn1 N1(C(=O)OC(C)(C)C)CCCOC(CNC(=O)NC23COC(CO)(C2)C3)C1 C1(O)(COC)CCN(C(=O)C(C2CC2)NC(c2cc(F)c[nH]2)=O)C1 CC1C(NC(=O)C(Cc2ccccc2)C2CC2)CCCN1C(=O)C(Cl)=CCl N1(C(c2cnc(C)s2)=O)CCCOC(CNC(c2ncccc2C(F)F)=O)C1 CC(N=c1[nH]c2c(c(=NCCN(CC(F)(F)F)CCO)[nH]1)CCCC2)C1CCOC1 CCC(CC)(C(=O)NCC=CCC(N1CC(C)(O)C1)=O)C(C)C c1(NC(C)=O)cccc(C(=O)N(C2CCN(C(=O)CC(F)(F)F)CC2)CCO)c1 C(=O)(CCCCCC(C)O)NC12CN(C(CSc3ccc(OC)cc3)=O)C(C1)C2 c1(C(C(N2CC(CC(C)N(C(=O)CCF)CCO)C2)=O)C)ccc2c(c1)OCO2 c1(OC)cc(N(C2CCNCC23CC3)C(=O)C(C)Br)cc(OC)n1 c1(C(=O)NC(CC=C)CNC(c2c[nH]c(=N)o2)=O)cc(Cl)c(F)cc1F c1(C(N2CC(N(C(c3cc(CC)c(Br)cc3)=O)C)C2)=O)cn2ncccc2n1 c1(-c2cn(C(C)C(=O)NCC(c3cnn(C)c3)=O)nn2)cc(O)c(F)cc1F N1(C(C2(C)C(C)(C)C2)=O)CCCCC(CNC(=O)CCn2cc[nH]c(=O)c2=O)C1 CCCC(CCC)C(=O)NC12CCC(NC(C3CCn4cncc4C3)=O)(CC1)C2 c1(OC(C)(C)C(N2CC(C)(C)C2C2CCOCC2)=O)ccnc(Cl)c1 CC1CCN(CCC(=O)NC2CCC(CNC(=O)CC(C)(C)O)CC2)CC1 C1(NC(CC(CC)C)=O)CCCC12CCN(C(c1cc(O)ccc1Br)=O)CC2 C1(NC(CC(C)n2cccn2)=O)CC2CCC(C1)N2C(C1CC2C(C1)C2(F)F)=O Cc1c(NC(C2CC3CC3N2Cc2cnc(Cl)nc2Cl)=O)cccc1O c1(C(N2C(C)(CNC(c3ccc(CF)cc3)=O)CCC2)=O)ncn2c1COCC2 C1(NC(C(C)N(C(c2cn(C(C)C)nn2)=O)CC)=O)CCC(OC)CC1 CC1(C)C(C(N2CCC(NC(=O)CCOCc3cccnc3)C2)=O)CCS1(=O)=O CC12CCN(CC1)CC2C(=O)NCC(O)CNC(=O)CSCC(N)=O C1(CNC(C2CC23CC3)=O)CC(C(F)(F)F)CN1C(=O)Cc1nc[nH]n1 C1(CC(=O)NC2(C(=O)NC(c3nccn3C)CC)CC(CO)C2)COCC(C)O1 Cc1cc(C(=O)NC2CC3CCC2N3C(c2nc(=O)n(C)[nH]2)=O)c2[nH]cnc2c1 N1(C(c2cc(C)nc(O)n2)=O)CCC(C2CCN(C(=O)CC(O)C3CC3)CC2)C1 C1(CNC(=O)C(F)CC2CCOC2)CN(C(C2CCCSC2)=O)CCCO1 C(=O)(C=C1SCC(=O)N1C)NCC(CC)NC(C1(C)CNC(=O)C1)=O N1(C(c2c(C)occ2)=O)CCOC(CNC(c2cc(C3CC3)ncn2)=O)C1 C1(C(=O)NCC(C)(O)CNC(C2CN(CC(C)C)C2)=O)(COC)CCNC1=O C1(F)(CNC(c2c(CC)ocn2)=O)CCN(c2nnc(C(N)=O)s2)C1 C1(C(N(CCNC(c2c(Br)noc2C2CC2)=O)CC)=O)CCN(C)C(=O)C1 N1(C(COCCCC#C)=O)CCC(F)(C(=O)Nc2cccc(CC)c2F)CC1 C1(C(N(CC2N(C(C=CC(CC)C)=O)CCC2)CC)=O)CN2CCC1CC2 CC1(C)COCC(C(=O)NCC2(C)CCN(C(=O)C3=CCCO3)C2)O1 c1(CSC)c(C(N2C3CCC2CN(C(c2ccoc2)=O)C3)=O)sc2ccccc12 c1(C(=O)NCC(C)CN(C)C(C23CSC(C2)C3)=O)ccnc(SC(C)(C)C)c1 C1(CNC(C(C2CC(F)(F)C2)OC)=O)CC2CCC1N2C(c1cc(Cl)on1)=O Cc1ccc(C(=O)NC2CCC(CCNC(=O)CCSCC(N)=O)C2)nc1C c1(C(=O)NCC2N(C(C3C(C(=O)OC)CCCC3)=O)CC2)cn2cccnc2n1 CC1(C)COC(C(N2CC(O)CC2CNC(=O)CCCc2ccsc2)=O)C1 C1(NC(C2=C(C)OCC2)=O)CC(Nc2ncc3ccnc-3[nH]2)C12CCOCC2 c1(NC(=O)Oc2cccnc2)ccc(OCCC(N2CC(C(N)=O)C2)=O)nc1 C1(OC)CN(C(=O)NC2(Cc3ccnc(Cl)c3)CC2)CC12CC2 N1(C(c2c(C)ocn2)=O)CCN(C(C2(CC(C)C)CCCC2)=O)CC12CCC2 N1(c2nc(C)n3c(c2)nnc3)CCN(C(C2CCC(C)CC2)=O)CC(C)(F)C1 C1(NC(CC(C)(F)F)=O)CCN(C(c2c[nH]cc2C(F)(F)F)=O)CC1(C)C c1(OC)c(C)cc(-c2cnc(CC(=O)NC3CCN(C)CC3)nc2)cc1C c1(OC)ncc(C=CC(N2CCC(CNC(=O)CCn3ccnc3)CC2)=O)cn1 C1(C(=O)NC(CC=C)CNC(=O)CCc2cc(C)no2)CC12CCCCC2 C1(CCNC(C(C)C2CCC2)=O)CCCN(C(=O)Cc2nncs2)C1 C1(C(N(CCOC)Cc2ccncc2)=O)CCCC2CCCN12 c1(C(N2C3CC(NC(=O)CCSC4CCCC4)(C3)C2)=O)occ2c1CCCC2 c1(C(N2CCC(N(CCC)C(c3cncn3C)=O)C2)=O)n[nH]c(CC)c1C CCCCC(C)CCC(=O)NCC1(F)CCCN(C(C2(C#N)CCCC2)=O)CC1 c1(C(=O)NCCC2CCN(C(c3ccn(COC)n3)=O)C2)ccc2nn[nH]c2c1 C(C1=NOC2CN(C(c3ccc(C4CC4)c(Cl)c3)=O)CC12)NC(CC)=O N1(C(c2nccc(C(=O)OC)c2)=O)CC2CCN(C(=O)CN3CCOCC3)C2C1 C1(CC(=O)Nc2ccc(NC(=O)CO)c(Cl)c2)(CO)CCCCCC1 N1(C(CNC(CCC)=O)=O)CC2CC1(CNC(c1cccc(CC(C)C)c1)=O)C2 C1(C)(C(N(CCC(C)NC(=O)C(C)(C)CF)C)=O)CNC(=O)C1 c1(C(=O)NCC23CCC(CC2)C3)cc2ccc(F)cc2s1.O=C1CC2(CC2)N1 N1(C(C(C(C(C)C)OC)O)=O)CCC2(C1)CN(C(=O)COC1CCOC1)C2 c1(C(CC)C(=O)NCC)ccc(OCCc2ccco2)cc1 C1(O)(C(C(=O)NC)N)CCN(C(=O)Cn2cc(C(=O)OC(C)(C)C)cn2)CC1.OC N1(C(c2nccc(C)n2)=O)CC(CNC(c2n[nH]c(C)n2)=O)OC(C)(C)C1 c1(CC(=O)N(C2(C(=O)N3CCCCCO3)CC2)C)ccc2c[nH]nc2c1 C1(C(N(C(CC)CNC(=O)CC2(C)CCOCC2)C)=O)CC2(C1)CC(O)C2 CCCCC(CC)C(=O)N1CC2CCC(CNC(C3SCCS3)=O)C2C1 c1(C(N2CC(C(C)NC(=O)C(C)(Cl)Cl)C2)=O)cccc2c1CCC(=O)N2 Cc1ccc(C(N2CCOCC2CN(C)C(=O)C2CC2)=O)cc1C1CC12CC2 c1(C(=O)NC(C(C)NC(c2n(CCC)ncc2)=O)C)c(C)cc(C)nc1S CC(C)(C(=O)NCCC(=O)NC1(C2CCCO2)CC1)n1ccnn1 CCCCCCCC(=O)N1CCC(CO)(NC(=O)Cc2cncn2C2CC2)C1 N1(C(c2c(OC)c(Cl)sc2)=O)CCN(C(C23CC(C)C2C3)=O)C(CO)C1 c1(C(=O)NCC2CC(NC(C3CCC(C)(C)C3)=O)C2)cnn2c1CCC2 N1(C(C2=NOC(C)C2)=O)CCC2(CCC2)C(NC(C2CCOC(C)(C)C2)=O)C1 C(=O)(CC(=O)NC1CC1)NC(CC)CN(C(C1(CN(C)C)CCCC1)=O)CC C1(C(N2C(CNC(=O)C(F)CC3CCC3)CCCCC2)=O)C2CCC3C(C2)CC13 N1(C(C2(SCC)CC2)=O)CCC(N(C(=O)CC(C)(C)N(C)C)CC)CC1 c1(C(=O)NCCCCCn2cc(C3(O)CC3)nn2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC(CNC(C(C)C)=O)(C)O)ccnn(C)c1=O C=CC1(C(=O)NCCC2CC2C2CC2)CCN(C(=O)C(C)C(F)(F)F)C1 C#CC1(C(N2CC3C(OC)C3C2)=O)CCN(C(C2CC(C3CC3)=NO2)=O)C1 C(=O)(CC(C(F)(F)F)NC=O)N(C(C)(CNC(C)=O)C(=O)OC(C)(C)C)C.C1(O)CCC1 c1(C(=O)Nc2cccc(NC(CS(C)(=O)=O)=O)c2)cccc2nccnc12 C(CCCCC(=O)NC1CCN(C(=O)Cc2[nH]cnc2C)CC1CO)OCC N(C1CCCc2cc(CNC(C3(C)CCC3)=O)ccc21)C(CC(C)(C)OC)=O C=CCC(CNC(=O)CC(C)NC(C)=O)NC(=O)C=CSC C1(NC(=O)C(F)(F)CO)CCN(C(C2(F)CC=CCC2)=O)CCC1(F)F N1(C(c2cc(C)sc2)=O)CCN(C(=O)CCN2CCC(F)C2)CC12CC2 c1(C(N2CCC2C2CCCCCC2)=O)ccc(C2(C(F)(F)F)CC2)c(Cl)c1O N1(C(CC(C)C2CCCO2)=O)CCC=C(CNC(C2CC(=O)NC2(C)C)=O)C1 CCC(C(=O)OC)C(=O)NC1CCN(C(C2C=CC=CC=C2)=O)CC1CO c1(C(=O)NCC2(F)CCN(C(C(C(C)C)(C)C)=O)C2)nnn2c1CSCC2 N1(C(C2C(OC)CCC2)=O)CCCC(NC(=O)CNC=O)C1CO C1(NC(C2CC(OC)C2)=O)CC2CCC1N(C(c1c(Br)ncn1C)=O)C2 N#Cc1cncnc1C(=O)NCC1CC(CNC(=O)C=C2CCCC2)CO1 C1(C2CC2)(CNC(C2CCC(C)C2)=O)CCN(C(c2cc(Cl)cc(F)c2N)=O)C1 C#CCC(C)(C)C(=O)N1CCC(C(C)NC(C2(n3cncn3)CC2)=O)C1 O=C(CC(F)(F)C(F)F)N1CCCC(N(c2ncc(I)cn2)CCO)C1 c1(C(N(C2CCN(C(=O)CC3CCC(O)C3)CC2)CCOC)=O)cc(C)cnn1 c1(C(N2CCC(CNC(COC)=O)CC2)=O)cc(Cl)c(F)cc1O Cc1cc2[nH]c(C(=O)NC3CC(C)N(C(=O)C(F)=CC4CC4)C3)cc2s1 Cc1cn2ccnc(C(=O)NCC(O)CCNC(=O)C3=COCCC3)c2n1 C1(NC(c2cccc(F)c2)=O)CC2CC1CN(C(c1coc3ccccc13)=O)C2 CC1CN(C(C2(F)CC=CCC2)=O)CC1c1cn(CCOc2ccccc2)nn1 C(C)(c1ccccc1C)=CC(=O)NCC1(O)CCN(C(CCC(=O)OCC)=O)C1 CC(CNC(=O)CCCc1ncco1)(CO)NC(C1CC(n2ccnc2)C1)=O Cc1c(C(=O)NC(C)CNC(c2cnn(C)c2C)=O)cccc1O C1(CC(N2CC(NC(CC3C(C)(C)C(O)C3)=O)C2)=O)CCC2(CC1)COC2 C1(C(=O)NC2C=CC(CNC(C3(OC)CC3)=O)C2)CC(C)(C)CCO1 Cc1ncoc1C(=O)NCc1cn(CC(=O)NCC2(N(C)C)CC2)nn1 N1(C(CCCOC)=O)CCCC(NC(c2oc(SC)cc2C)=O)C1C C1(C(N2CC(NC(c3n[nH]c(C)c3O)=O)C(C)CC2)=O)CC2CCCC(C1)C2 c1(CCC)ccc(C(=O)NC23CCC2CN(C(=O)C(C2CC2)OCC)C3)cc1N Nc1cc(C(N2CCCC(NC(C34CC(CN3C3CC3)C4)=O)C2)=O)cc(O)c1 N1(Cc2c(OC)ccc(C)c2)CCC2(CCN(C(=O)CN3C(=O)CSC3=S)C2)C1 N1(C(C23CC(NC(=O)CC4C=CCCC4)(C2)C3)=O)CCC2CC1CO2 C(=O)(C(=O)N=c1cc(-c2ccc(C#N)cc2)[nH][nH]1)c1ccc(C=C)cc1 N1(C(CCC(C)N(C)C)=O)CC=C(C(=O)NCC2(C)CCCC(=O)N2)CC1 Cc1cccc(-c2cccc(C(=O)NC3(C)CN(c4ncncc4I)C3)c2)c1 c1(C(=O)NCC2CCCC2NC(=O)CCc2ccccc2F)cc(F)cc(Cl)c1 C(=O)(C1=CCCCC1C)NC1CC2(C(NC(c3cnc(CCC)s3)=O)C2)C1 c1(C(=O)NC2(C)CC(NC(=O)C3=CCC3)C2)ccc(Br)cc1[N+](=O)[O-] C1(O)(C(N(CCCCN(C(c2nn(CC)c(O)c2)=O)C)C)=O)CCCC(C)(C)C1 C1(Nc2nccc(C)n2)CCN(Cc2c(C)cccc2C)CC1O c1(C(N2CC(COC)N(C(=O)Cc3nnc(C)o3)CC2)=O)c(Cl)ccc(F)c1C C1(NC(c2c(Cl)cc(C)s2)=O)CC2CCC(C1C)N2C(c1nc(C)n(C)n1)=O n1(CCC(=O)NCCC2CCC(NC(c3ccc(O)cc3)=O)C2)ccccc1=O O=C(CC(C(F)F)c1ccc(F)cc1)NCCC1CCCC2CC12 C1(C(=O)NCC2CCC=CCC2)CC=CCN1C(c1ncccc1O)=O N1(C(c2cn(CC)nn2)=O)CCCC12CCCN(C(=O)CC1C=CCC1)C2 C1(C2CC2)(C(N(CCN(C(C(CC#C)O)=O)C)C)=O)CCOCC1 C1(COC)CCC(N=c2nc(NCCC3CCC3)c3c([nH]2)CCS3)CC1 N1(C(c2c(SC)nc(O)nc2C)=O)CCC2(CCC2CNC(=O)CC(C)F)CC1 c1(OC)ccccc1C(N1CCCCC1CCNC(c1ccoc1Br)=O)=O c1(OCC(C)(C)C)ccc(C(=O)NCCC(C)(C)NC(C2CC(O)C2)=O)cc1 c1(NC(C2SCCN(C(C#C)=O)C2)=O)ccc(F)c(COC)c1F CCC(C)(C)C(O)C(=O)N1CC2(CC2)CC1C(=O)NC(c1nccs1)C C(=O)(C(F)CC(C)C(=O)NC(C)(C)C)N(C)CCNC(C1(C#N)CCC1)=O c1(C(=O)NCC2CC(NC(C(CCC)N(C)C)=O)C(O)C2)nc2cccnc2s1 CCCCC(C)(F)C(=O)NC1CCCC1C(=O)NCCc1cscn1 c1(C(N(CCCNC(C(C)=C2CCC2)=O)C2CC2)=O)ccc2nc(CO)[nH]c2c1 C(CCN=c1nc2ncn(C)c2c(NC2CC(OC)C23CCCC3)[nH]1)NCC CCCC(F)C(=O)NC(Cn1ccnn1)C(N1CCCC(CN(C)C)C1)=O Cc1cc(Br)c(C(=O)NC2CC(NC(c3cncn3C)=O)C2)cc1Cl c1(COCC(=O)N(CCNC(C23C=CC(CC2)C3)=O)CC)nc2ccccc2s1 c1(NC(C(N2C(CNC(C=CCOC)=O)C=CC2)=O)C)ccccc1-n1ccnn1 C1(CNC(C(C)(C)Cc2cnn[nH]2)=O)CC2CN(C(=O)C3=CCCO3)CC12 C1(CNC(C=CC(CC)=CC)=O)CC(C)N(C(c2cc(CC)c[nH]2)=O)C1 N1(C(C23CC(NC(c4scc(C)c4Cl)=O)(C2)C3)=O)C2CCC1CC(F)C2 C(C(C)(O)C(=O)N1CCCC(n2cc(C(C3(OC)CCCC3)C)nn2)C1)OC O=C(N=c1ccc(Br)n[nH]1)NCCOCCNC(=O)NCc1cc(Cl)sc1Cl CC(C(=O)NC1CCCN(C(=O)CC(=O)NCC(F)(F)F)C1)C(F)F N1(C(c2ncc(C(N)=O)nc2)=O)CCC2(CCN(C(c3cccc(Cl)c3)=O)C2)C1 c1(C(=O)NC(CC)CN(C(=O)Cn2ccc(C)n2)CC)cccc2oc(O)nc12 c1(C(N(CCC)CCOC)=O)ncccc1Cl.c1(C(=O)OCC)cc(CO)oc1C Cc1nc(C(=O)NCC2CN(C(=O)COCC(C)C)CCC2C)c2ccccn12 N1(C(C(CC(F)F)N(C(C(CC(C)C)O)=O)C)=O)CC2(COCC(=O)N2)C1 C1(NC(CCCC#C)=O)CCN(C(=O)C=C(C)c2ccsc2)CC1F C12(C(C)NC(C3C(C(C)NC(C4CC(=C)C4)=O)C3)=O)CCC(CC1)C2 c1(C(=O)NCC(C2CC2)NC(C(=O)NCC)=O)cc(C(F)(F)F)ccc1Br c1(C(=O)NC2(C(=O)NCC3CCN(C(C4CC4F)=O)C3)CC2)ccc(F)c(Cl)c1 N1(C(c2nnn(CC)c2C)=O)CCN(C(=O)C=CCOCCOC)CC1C Cc1c(-n2cc(CNC(=O)CNC(=O)CC(C)C(F)F)nn2)cccc1N Cc1cc(F)c(CC(N2CCCOC(CNC(=O)CC(=O)N(C)C)C2)=O)cc1F Cc1ccccc1CNC(=O)C(N1CC2CC2C1)C1CCCC1C c1(C(=O)NC(CC=C)C(=O)NCC2CCOCC2)c[nH]c2ccncc12 C1(C)(NC(C(C(=O)OC)C)=O)CCC(NC(=O)Cc2ccc(C)o2)CC1 c1(CNC(c2ccc(O)nc2)=O)ccc(CNC(c2ccc(CO)cc2)=O)cc1 C(=O)(CCS(N)(=O)=O)NCC1(C(=O)NC(C)CC(F)(F)CC)CC(=C)C1 C1(C(N(CCCNC(C=CCCC(C)C)=O)C)=O)COCCC1C C1(C(=O)NCC2CCC(F)C2)(NC(C(CC)OC)=O)CCCCCC1 N1(C(c2nn(CC)c(O)c2)=O)CCN(C(=O)Cc2ccoc2C)C2CCC12 C1(C(=O)NC(C(=O)OCCC)CC)CC2(C1)CC21CCC1 n1(CC(=O)NCC#C)c(-c2ccsc2)nc2ccccc12.C12CCN(CC1)C2 c1(C(N2CC(C)C(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)cnc(Cl)c(F)c1 c1(C(N2CC(F)(F)CC2CC(N)=O)C(=O)NC)cn2cc(F)ccc2n1 N1(C(C(C2CCCC2)OC)=O)CCCCC1CCC(=O)NCC1CCC1(F)F N1(C(CSC)=O)CCCN(CCNC(c2ccccc2C2CC2)=O)CC1 C1(NC(C(Cc2c(C)nc[nH]2)O)=O)CCCC12CN(C(=O)CCNS(C)(=O)=O)C2 S(=O)(=O)(c1cccs1)N1C(C)(C(N2CC(C)C(O)C2)=O)CCC1 c1(C(N2C(C(=O)NCCS(N)(=O)=O)CC(F)C2)=O)cc(Br)cc2cn[nH]c12 c1(C(=O)OC)cc2n(c1)CCN(Cc1ccc(CN(C)C)o1)C2 c1(C(=O)NCC2(NC(=O)CCC=CBr)CCC2)cccc2c1C(=O)NC2 C1(O)(C(C)CNC(c2cocn2)=O)CCN(C(=O)CCOc2ccccc2O)C1 C1(NC(c2cccc[n+]2[O-])=O)C2CCC1N(C(=O)C1=CCC1)C2 N1(C(=O)Cc2ncsc2Cl)CC2(CCN(C(c3c(F)cccc3F)=O)CC2)C1 Cc1cc(O)nc(SCC(=O)OCC2CCC(C)(C(C)(C)C)C2)c1C#N C1(C(N2C(C)CC(CNC(c3c(CC)n(C)nc3)=O)C2)=O)CC2CCC(C1)O2 c1(N2CC3C(NC(C(CC)(C)C)=O)C3C2)nc(C)c(C#N)cc1Cl c1(C(CNC(=O)Nc2ccc(N(CCC)C)cc2)(C)C)c(C)nn(C)c1Cl N#Cc1cc(F)c(NC(C2CC23CN(C(=O)CC2(O)CCC2)C3)=O)cc1Cl N1(C(CC)=O)CCN(C2CCCC2NC(=O)CCN2CCCC2)CC1 c1(CC)cn2c(C(=O)NC34CCC(C3)N(C(c3nncs3)=O)C4)cccc2n1 N1(CCNC(c2nccc(=N)[nH]2)C)CCC(c2ncco2)CC1 c1(OC)cnc(F)c(C(=O)NCC(C)(C)NC(=O)CC2CC3(CC3)CO2)c1 N1(C(CCCCC=C)=O)CCCC1C1CCCCN1C(=O)CN(CC(=O)NC)C c1(SC(C)C)ccc(C(=O)NCCOCCNC(=O)CSS(C)(=O)=O)cc1 N1(c2cc(C(=O)NC(C3CC3)C3CC3)ncn2)CCC(CC(O)C(F)(F)F)CC1 C12(CNC(CCN(C(c3ccncc3O)=O)CC)=O)CC(CN1C)C2 c1(C(N2CC(NC(C3CC(OC)C3)=O)C(C)C2)=O)cc(C)c(C)nc1C C1(CNC(C(CC=CC)C)=O)COCCN(C(c2ccoc2C2CC2)=O)C1 C1(C(=O)NC(C2CN(C(C3(Sc4ccccc4)CC3)=O)C2)C)CCCOC1 CCCCC(CNC(C1CC(C(F)(F)F)C1)=O)NC(C1(C)CC=CC1)=O c1(C(=O)NC(CCOC)CNC(c2cc(F)c[nH]2)=O)cnc(OCC2CC2)cn1 C1(C(=O)NCc2nccc(C(=O)NC(C#CC#C)(C)C)c2)CCCCC(=O)C1 C(=O)(C#CC1CCCCO1)N1CCN(C(c2cc(OCC)n[nH]2)=O)CC1 C1(CCNC(=O)Cc2cnco2)CC(F)(F)CN1C(=O)CC1CCCCC1 CCC(CCOC)C(=O)NCC1CC(OC)CN1C(c1nonc1N)=O N1(C(COCCC)=O)CCOC(CNC(c2ccn(C(C)C)c2C)=O)C1 N1(c2nnc(-c3nc(COC)sc3)n2CC(C)C)CCCC(C#CBr)CC1 c1(C(=O)NC2C(CC(=O)N(CCN(CC)CC)C)CCCC2)cc(C)nc(C)c1 CC1(F)CN(C(C2(NC(C3CNC(=O)N3)=O)CCSC2)=O)C1 c1(C(=O)NCC(CC(C)C)NC(=O)C=C(Cl)Cl)cc(F)c(O)c(F)c1 c1(C(=O)NCC2N(C(C(C=C)C)=O)CC(F)C2)ccncc1N=[N+]=[N-] Cc1cc2[nH]c(C(=O)N(C3CC4CCC(C3)N4C(=O)C=CC(N)=O)C)cc2s1 C12(C(=O)NCC3CC(F)(CNC(=O)C=C4CCOCC4)C3)CCCCC1C2(F)F S(=O)(=O)(C=Cc1ccccc1)NC(c1cc(Cl)cc(F)c1Br)=O C1(C(=O)NC23C(CN(C(c4cccc(CC)n4)=O)C2)C3)Cc2c(C)cccc2O1 c1(CNC(=O)NC2C(OC(C)(C)C)C2)ccc2nnn(O)c2c1 N1(C(c2cnn(CCC)c2C)=O)CC(NC(C2CC2F)=O)C2(CC2)C1 c12cnn(C)c1C(=O)NC2.n1(CC)cnc(C(=O)NCCCc2ccccc2)c1 CC1CCC(CCC(N2CC(O)(CN(C)C(c3ccsc3)=O)C2)=O)O1 CN1CC(C(=O)NCCCN(C(=O)C(c2ccccc2)C2CC2)C)CC1=O c1(C(=O)NCC(NOC)=O)ccc(Nc2cnc(OC(C)C)cn2)cc1 CC(CC(=O)NCC(Cl)Cl)C(C)(C)NC(=O)C(c1cnn(C)c1)C c1(C(N(CC(CC)NC(c2ccc(CC)cn2)=O)CC)=O)ccc2c(n1)CCC2 C(CCCCC(=O)NCC12CC(CO1)N(Cc1cc3sccc3[nH]1)C2)NC(N)=O c1(CCC(=O)NC(CNC(COCCOCC#C)=O)(C)CO)cccc(C)c1 c1(CNC2CC(C(N3CCN(S(C)(=O)=O)CC3)=O)C2)cccc2ccccc12 C(=O)(CC1=Cc2ccccc2C1)N1CCN(C(C=CC(C)C)=O)C(C(F)F)C1 N1(C(c2nc(C(C)C)sc2)=O)CC2CC(NC(=O)C=CBr)C2C1 S(=O)(=O)(c1cc2sc(=NC3COCC3C)[nH]c2cc1C)N1CCC(C(C)O)CC1 Cc1nccn1CCNC(C1CC(C)N1C(=O)Cn1cccn1)=O c1(C(=O)NC2(CNC(c3cc(C(=O)OC)on3)=O)CCC2)cccc(Cl)c1Cl c1(C(=O)NC(C)CC2CN(C(c3cccc(F)c3Cl)=O)C2)cc(Cl)ccc1F C=CCCCC(C(=O)NCC1CC2CCC2C1)NC(=O)C(C)N=[N+]=[N-] c1(NC(C2CC(=C)CN2C(c2nc(C3CC3)cs2)=O)=O)ccc(Br)c(Br)c1 CC(C)(C)C(C#N)C(=O)NC(C(N1CC(O)(C2CC2)C1)=O)C1(O)CCC1 C(c1cccnc1)=C(C(=O)NC(C)C(CO)C(=O)OC(C)(C)C)F.CC1C(=O)N1 c1(C(=O)NC(CN(C(=O)COCCC(C)C)CC)C)cncc(C(C)C)c1 C1(CCNC(Cc2nc(C)sc2C)=O)C(C)CCCN1C(=O)Cc1cn(C)nn1 Cc1cc(C(=O)NCC2CCCCC2NC(C2CC23CCCCC3)=O)nc(C)n1 n1(CC)c(-n2nc(COCC(F)(F)F)nc2CO)nc2ccccc12.SC(F)F C12(C(=O)NCC(C)CC(C)O)CC(C)(CN1C(=O)C=CC1CCC1)C2 N1(C(CC(CC)C2CC2)=O)CCn2ncc(CNC(=O)C3=COCCC3)c2C1 c1(C(=O)NCC2C(C)(C)C(NC(=O)CCN3CCOCC3)C2)cccc(O)c1Cl c1(Cc2ccc(NC(c3ccc(O)c(F)c3)=O)cc2)ccc(Cl)cc1Cl O=C(C1CCc2scnc21)NC1CC(NC(C2(CCF)CCC2)=O)C12CCC2 Cc1cc(Cl)c(C(=O)NC2(CF)CCN(C(C3(C)CCCC3C)=O)C2)cn1 C(=O)(C1=C(CCCCC2CC2)N(CC)C(=O)NC1c1cncn1CC)OCC Cc1ccc(CC2CCCC2NC(=O)NOCC(O)C(C)C)cc1 c12csc3ncn(c(=O)c13)oc2=O.[N-]=[N+]=Nc1ccc(Cc2ccccc2)cc1 S(=O)(=O)(CCN=C(NCC(C)(C)C1CCCC1)N(C)CC1CC1)NC c1(C(N(C(CNC(C(COC)O)=O)C)C)=O)cc(S(=O)(=O)N(C)C)oc1C C1(CC(=O)NC2(C(=O)NCC)CCCC2)CCCCN1C(c1cnsc1)=O N1(C(C(C)O)=O)CCCC(CCCNC(c2ccc(C3CC3)cn2)=O)C1 c1(CNCC(C)N(C(CCSC)C(=O)N(C)C)CC(C)C)ccc(Cl)c(Cl)c1 CN1C(=O)CCC1C(=O)NCC=CC(=O)NC1CC(CO)C1(C)C N1(c2nc(C)nc3c2c[nH]n3)CCc2cc(NCc3cc(Cl)c(Br)s3)ccc2C1 c12ncccc1C(=O)NC2.CC1CCCC1CC(=O)N(CCO)CC1CNC(=O)C1 C1(NC(C=CC)=O)C2CCN(C(c3ccc4cnoc4c3)=O)CCC12 c1(C(=O)NC2(CNC(COc3ccc(C)cc3)=O)CC2)cc2c(C)cccn2n1 c1(CN(CC(=O)NCC(=O)OC)C)cscc1Br c1(OCC(=O)NCC(CN(C)C(c2cccc(Cl)c2N)=O)O)ccc(F)c(Cl)c1 N1(C(C(=C(C)C2CC2)F)=O)CCC2(CC1)CC(NC(=O)C(C)OCCN(C)C)C2 C1(O)(CNC(C(C=CC)O)=O)CC2CCC(C1)N2C(c1ccncc1C(F)F)=O c1(C(=O)NC2CCCN(C(CC=CCC)=O)CC2F)c[nH]c2ccc(OC)cc12 C=CC(C)(O)CC(=O)N1CC2CC2(CNC(=O)Cn2nnc(C(=O)OC)c2N)C1 C1(NC(C2CC(C)=C(C)CC2)=O)CN(C(c2coc(Br)c2)=O)CC2(CC2)C1 CC1(C)Cc2ccc(C(=O)NCC3(O)CN(C(C4COC(=O)C4)=O)C3)c(O)c2O1 Cc1cc(OCC(N2CCCC(NC(c3ncc(F)cn3)=O)C2C)=O)cc(C)c1 c1(COC)ccc(NC(c2oc(C3CCOCC3)nc2C#N)=O)c(F)c1 C(=O)(CCNC(c1cscn1)=O)NCCN(C(=O)COCC1CC1)CCC C#CC(CC1CC1)CN=C(NC(C)C)N1CCCC1.CS(C)(=O)=O N1(C(C2C(CC)C2)=O)CC(O)(CCNC(=O)CSc2cccs2)C1 CCC(C)C(=O)NC(C)COCC.C12(CCCC1)C(=O)N2 C(=O)(C(CCC(C)C)NC(c1ccnn1COC)=O)Nc1ncc(CC)s1 c1(C(N2CC(CNC(CCC(=O)NC)=O)C2)=O)ccc(OC)c(Cl)n1 CC1(C)CC(CC(N2CC(OCCNC(C3CC4(CCCC4)C3)=O)C2)=O)CCO1 c1(NC(=O)NCC(n2cc(C3CCOC3)nn2)C)ccc(-c2nncn2C)cc1 c1(C(c2nnnn2C2CCCCC2)NC(c2cnc(Cl)s2)C)nc(C(C)(C)C)cs1 c1(C(N2CCC(N(CC#C)C(C3OCCOC3C)=O)CC2)=O)cc(N)cc(F)c1 c1(CC(=O)NCC(CC2CCCC2)C(=O)O)ccc(F)cc1.C12CC1C2 CN1CCCC1CC(=O)N(C1(C(=O)NCC2(N(C)C)CC2)CC1)C O=C(C1CCc2nccn21)NCC1(CNC(C2CC23CCOCC3)=O)CC1 C1(C(=O)NC2CN(C(CCCOC)=O)C(C)CC2)Cc2cncn2C(=O)N1 C1(C(=O)NCCC2N(C(C(CC(N)=O)O)=O)CCOC2)CCc2nnc(O)n2C1 C(=O)(CS(=O)(=O)CCO)N1C(C)CC(NC(=O)CN2CCN(C3CC3)C2=O)CC1 CC1COC(CNC(c2ccc(CNC(C3(CC4CCC4)CC3)=O)o2)=O)C1 Cc1csc2cncn12.N1(C(C(N2CCC(C=O)C2)=O)=O)CC(CO)C(O)C1 CC1CN(C(C2CCCCCC2C)=O)CCN1C(=O)CCC(C)(F)F c1(C(N2C3CC(CC(NC(C(C)OCC#C)=O)C3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(NC(C2N(C(CC(=O)NCC)=O)CC(F)(F)C2)=O)CN(C)C(=O)C12CC2 C#CCC(CC(F)F)C(=O)N1CCC(C(N2CCC3CC23)=O)C(C)(C)C1 C1(NC(CC2CC(NC(C(C)n3cncn3)=O)C2)=O)CC(F)(F)C1(C)C C(=O)(C(=O)N=c1cc(C(F)F)o[nH]1)c1nc(C2C(C)(C)CN2)on1.c12cccc(c1)N2 C(C1CN(C(C2CCC2C(N)=O)=O)CC1C(N1CCSCC1)=O)=CC n1(CC)ncc([N+](=O)[O-])c1C(=O)NCC(O)CNC(=O)CC1(CSC)CC1 N1(C(C2(CC#C)CC2)=O)CCC(CCOC)(NC(=O)C(c2ccccc2)OC)C1 N1(C(c2cc(C(C)=O)oc2C)=O)CCC2CN(C(=O)CC3CC4(CC4)CO3)C2C1 N1(C(C(C)Cn2cccn2)=O)CCn2nc(C(=O)N(C3CCC3)C3CC3)cc2C1 C1(C2CC2)(COC)CCN(c2nnnn2-c2ccc(F)cc2C(F)(F)F)C1 N1(C(c2n(CCC)nc(C)c2)=O)CC=C(CCNC(C2CC(C)(C)C2)=O)CC1 c1(OC)cc(F)c(C(=O)NC(CNC(=O)C(C)(C)N(C)C)C(C)(C)C)c(F)c1F c1(C(=O)NCCCCCNC(COCCC=C)=O)cncc(C)c1Cl N1(C(C(CCC)NC(N)=O)=O)CC2CC(NC(C3C=CC=CC=C3)=O)C(C2)C1 CCCCCC(C)(C)CNC(=O)C(C1CCN(C(C2CCC(CC)CC2)=O)C1)C C#CCC(C)(C(=O)N1CCN(C2CC2)C(C)C1)NC(c1cc(C(C)C)no1)=O C1(NC(=O)CC2CC3CC3C2)C(CN=c2[nH]ncs2)CCC12CCC2 c1(C(=O)NCCC(C)N(C(C(F)OC)=O)C)cccc([N+](=O)[O-])c1Cl c1(CC(N2CC(N3C(=O)CC(CNC(C(N)=O)=O)C3)C2)=O)cc(F)cc(Br)c1 N#Cc1cc(Br)ccc1NC(C1CCCN(C(C2CC(O)C2)=O)C1)=O C1(O)(CCNC(c2c(CC)non2)=O)CCN(C(=O)CCC2CCCC2)C1 c1(CNC(=O)NCC(=O)OCC)ccc(OC)c(Br)c1N Cc1cccc(C(=O)NC(C(=O)NC2COCC2CO)C(C)C)c1O CCC(CC(=O)NC1CCN(C(=O)Cc2ccns2)C1C(C)C)SC c1(CNC(=O)CC2CCCN2)c(O)cccc1Cl C12(C(=O)NCCC3CC(NC(C(CCC)(C)CC)=O)C3)CC(C)(C1)OC21CCC1 C(C(CO)CC(C)(C)C)NC(=NCCOCC)NC1CCCN(CC)C1 Cc1ccnc2ccc(C(=O)NC3CCC3NC(=O)CCCS(C)(=O)=O)cc12 c1(C(N2CCC(CCNC(C3N(N=O)CCC3)=O)C2)=O)csc2c(O)ccnc12 CC(CNC(=O)C(CC1CCC1)NC(c1csnc1Cl)=O)N=[N+]=[N-] Cc1ccc(Cl)cc1C(=O)NC(Cc1ccccc1)CCNC(=O)C=CC1CC1 C1(CC)CN(C(=O)CC2CC2CNC(=O)Cc2cn(C)cn2)CC(=O)N1 N1(CCN(C)C)CC2CC(CN(C(=O)Cc3ccc(OCC(F)F)nc3)C)CC1C2 C1(NC(CCC(=O)NCC)=O)C2CCC1N(C(=O)Cn1nnc(C3CC3)n1)C2 Cc1cnc(C(=O)NCCCN(CCO)C(c2cnc(C(C)C)o2)=O)cn1 C(=O)(C(C(C)C)NC(=O)C(C1CCCO1)SCc1ccc(CO)o1)N(C)OC c1(C(N2CC(NC(c3n(C(C)C)ccc3)=O)C2)=O)cc2[nH]ccc2s1 N1(C(C2(F)CC(C(=O)OCC)C2)=O)CCOC(CNC(=O)CC2(C)CCCC2)C1 NC(=O)CCCC(=O)N1CC2C(CNC(=O)COC(F)(F)F)C2C1 N1(CCO)C(=O)N2CCCC2(C)C1=O.CCCCC(COC(C)C)n1nnnc1CC C1(NC(c2csc(C(F)F)c2)=O)CCC2CCN(C(c3ccc(F)cn3)=O)C1C2 C1(N(C)C(c2ccccc2Cl)=O)CN(C(=O)COC(C)(C)C)C(C)(C)C1 N1(C(CC2CC(=C)C2)=O)CC(CNC(=O)C(F)=CCCN2CCOCC2)C(C)(C)C1 CC(C)C(F)C(=O)NCCCN(C(=O)CCC1CC(C)(C)CO1)CCO N12CCN(CC1)c1cc(ccn1)NC2=O.C1(NC(C)C)CCOC(C(F)F)C1 c1(NC(C2CC3CC3N2Cc2cnc(Cl)cn2)=O)nccc(Cl)c1Cl c1(C(=O)NC(CC(C)NC(COC)=O)C)ccc(C)n1C c1(C2C(NC(C(=O)NCC(CN)OC)=O)C2)ccc(F)c(Cl)c1 C1(NC(C2CCCN(C(c3nccc(C)c3)=O)C2)=O)C2CCC(C2)C1CO c1(C(N2CC(C)C(CNC(c3ccc(C(N)=O)s3)=O)C2)=O)cn2ccccc2n1 C1(SCC)CCC(c2c(OC)cccn2)CC1.c1(NCCNC=O)ccnc(Cl)c1 N1(C(C2C(C3C(C)C3)C2)=O)CCC(N=c2[nH]nc(CC(F)(F)F)s2)(CO)CC1 N1(C(C)=O)CCCC1C(=O)NC(C1CCCC1)CN(C(=O)C(C)(C)C)C(C)C Cc1cc(C(=O)NC2(CO)CCCN(Cc3ccncc3Cl)C2)c(C)cc1O C(CCC(C)C(=O)NCC(C1CCCN1C(=O)Cc1cncn1C)(C)C)OC C1(CCC(=O)NC(C)Cc2cccnc2)CCCCN1C(c1csc(Cl)n1)=O C(C(=O)NCc1cccs1)(C(C)O)NC(Cc1c(C)scc1)=O C1(CNC(C2CCN(C)C2)=O)C2CCC(C2)N1C(C1(S(C)(=O)=O)CC1)=O C1(C)(C(=O)NCC(C)CN(C)C(c2conc2C2(C)COC2)=O)CCCCO1 Cc1nn(C)c2c(NCC3CN4CCC3CC4)nc(=NCC3CCC3(F)F)[nH]c12 C1(NC(COCC#C)=O)CC(CNC(c2ccc(CF)cc2)=O)C1(C)C N1(C(C=CC)=O)CC(CNC(c2cc(COCC)ccn2)=O)OC(C)(C)C1 Cn1nc(CC(=O)NCC2CCN(C(=O)CCc3cncs3)C2)cc1C(N)=O Cc1ccc(CCC(=O)NCC(=O)N(C(c2cnccn2)C2CC2)CC2CC2)cc1 C(CCNC(c1cn(C2CC2)nn1)=O)(C(=O)OC)OC.C12C=CC(C1)CC(=O)N2 N1(C(c2c(C(C)C)onc2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC(C)(F)C1 C(=O)(C(C(C)(C)C)c1cc(F)cc(F)c1)NCC(C)NC(=O)C(F)F N1(C(c2c(OC)ccs2)=O)CCC(NC(c2ccnn2C)=O)C1C(C)(C)C C(C(=O)N(CC(=O)NC)C)(C(C)C)c1nnc(CC)s1 O=C1OCC2CN(C(=O)C(N3CC4CC5(CCC5)C4C3)=O)CCN12 C1(NC(C(c2cc(=N)[nH][nH]2)(C)C)=O)CC=C(C(=O)NC2Cc3cscc3C2)C1 c1(C(N(CCN(C(C2C(CC)N(C)CC2)=O)C(C)C)C)=O)ccc(N)cc1Cl C1(CNC(C2(C#C)CC2)=O)CC12CCN(C(C1CN3CCN1C(C)C3)=O)CC2 C(=O)(C1=NNC(=O)C1)NC1CC(CNC(CCCn2c(C)cc(C)n2)=O)C1(C)C c1(CONC(C2CC(N)C2)=O)csc(Cc2ccccc2)n1 C(N=c1nc2c(cnn2C)c(NC(c2ccoc2)C)[nH]1)C1CCN(CCOC)C1 C1(C(=O)NCC2(OCC)CCC2)CNC(=O)CN1C(=O)C(C)CC1CC1 C1(C(N(CCOCC)CCSC)=O)CC(OC)CN1C(c1nnsc1C)=O c1(C(=O)NC2CN(C(C3C(C)(C)CC3)=O)CC2C(F)F)nccc2occc12 C(=O)(CCCCCCn1cc(CN2CCCC2)nn1)NC1(C)CC(O)C1 Cn1cc(C(=O)NCCNC(c2ccc(N3CCCC3)cc2)=O)ncc1=O C1(CC)C(C(=O)NCCc2ccccc2)CCN1C(=O)C(=Cc1cnn(C)c1)C Cn1cc2c(C(=O)NC34CCC(C3)N(C(=O)COC3CC3)C4)cccc2n1 C1(C(=O)OC)C(C)CCCN1C(c1ncc(F)cc1C)C(=O)NCCCC1CC1 S(=O)(=O)(c1ccc(S(=O)(=O)Nc2ccc(N(C)C)cn2)cc1)NC(C(C)O)=O CC(C)CC(O)C(C)C(=O)Nc1cncc(C2CC2)c1.C1(C)(C)CC(=O)N1C CC(C)CC(CC(=O)NC1COCC(C)(C)C1)NC(c1cccc[n+]1[O-])=O c1(C(=O)NC(c2cnn(C)c2)C(=O)NCCC2(C)CC2)cn(C2CC2)cn1 N1(C(C2CC(=C)C2)=O)C2CCC1(CNC(c1cnc3n1CCS3)=O)CC2 c1(CCC(=O)NC(C(C)NC(C2CNC(=O)N2)=O)(C)C)cccc(F)c1F n1(CC)c(C)nn(CC(N2CCOC(CN(C(=O)C(C)OC)C)C2)=O)c1=O N1(C(c2c(Cl)ccc(OC)c2)=O)CC2CCC1CN2C(=O)C(C)OC n1(CC(=O)NCC(CNC(COCC)=O)CO)cccnc1=O CCCS(=O)(=O)C(C)C(=O)NCC(O)CNC(c1c(N)sc2c1CCC2)=O S(=O)(=O)(CC(=O)NCC(F)CNC(=O)C(C)NC(C)=O)NC CCC(CC(C)C)C(=O)N1CCC12CN(C(c1nonc1N)=O)C2 C(=O)(C(C)CC(F)(F)F)N1C(CNC(CS(CC)=O)=O)C2CCC1C2 C12(NC(CCCC=C)=O)CCC1CN(C(c1ccc(CN(CCC)CC)o1)=O)C2 C12(CNC(CCCCSC)=O)CCC1CCN2C(=O)CSCCN1CCCCC1 c1(C(=O)NC2(CCCNC(CCC(=O)N(C)C)=O)CC2)ccn2ccccc12 C1(CNc2cnn(C(C)C)n2)N(C(=O)C(N2C(C)CCC2C)C)CCCC1(C)C C=C(C)CN=C(NCC1(OC(C)C)CCOCC1)NC1CCSC1 CC(C)C(O)C(F)(F)C(=O)NCCN1CCCN(C(=O)Cn2nccn2)CC1 Cc1nc(C(N2CC(NC(C3CCN(C)C3c3ccccc3)=O)C2)=O)c(=O)[nH]c1C C1(C)(C(=O)NCC(CNC(CCOCC(C)C)=O)(C)O)CCCNC1=O c1(C(N2CC(O)(C(C(=O)NC3C=CC(C(=O)NC)C3)F)C2)=O)ncc(C)cc1C C1(NC(C(=O)N(C)C)=O)COCCN(C(=O)Cc2ccccc2NC(N)=O)C1 N1(C(CC(C)(C)CNC(c2cnccn2)=O)=O)CCC2(CCCOC2)C1 N1(CCN(C(C(C)NC(C2CCC2)=O)=O)C)CCN(C(=O)CC(C)(F)F)CC1 C1(COC)(NC(=O)Cc2nccs2)CN(C(=O)C(c2ccc(C)s2)C)C1 c1(C(N2CCC(CCNC(CSCC=C)=O)C2)=O)ncccc1-c1ccccc1 N1(C(C(C=C)O)=O)CC(C)(C)OCC1CNC(c1c[nH]c(=N)cc1C)=O c1(C(N2CCC3(NC(CCNC(=O)NC)=O)C(C2)C3)=O)c(F)ccc(Cl)c1N C(=O)(CC(C)C(F)(F)F)N1CC(C(=O)NCCC(C)SC)(CC)C1 CC(C#N)C(=O)NC1(CN(C(=O)CN(CC(C)(C)C)C)C)CC1 C1(C(N2CCC(C(=O)OCC)(OS(C)(=O)=O)CC2)=O)CCc2nc(CC)cn2C1 N12CCN(CC1)CC2=O.c1(C2(NC(N)=O)CCC2)ccc(Br)s1 N1(C(c2c[nH]c(C)c(Cl)c2=O)=O)CC(CNC(=O)C(=O)NC(C)C)CC(C)(C)C1 Cc1nc(C(F)(F)F)oc1C(N1CC(N(C)C(C2CCC2C)=O)C1)=O c1(C(N2CC(n3cc(-c4cnn5ccccc45)nn3)C2)=O)nc2cc(F)ccc2s1 C(C(C(=O)N1CC=CC1CNC(C1CCOC1C(C)C)=O)N(C)C)OCC C(=O)(CCCC(F)F)NC1CCC(C)(CNC(c2ccc(C(N)=O)o2)=O)C1 c1(C(=O)NC2CN(C(=O)CCn3cncn3)CC2F)ccc2cccc(F)c2n1 N1(C(C(F)=CCC)=O)CCC(F)(C(=O)NCCOc2ccccn2)C1 c1(C(c2nnnn2CCC2CC2)NC(C)C)nnc(C)n1C C(CC)(CC)(CCNC(=O)C(C)(O)C1CCC1)NC(C(CCC)NC(C)=O)=O Cc1ccc(F)c(C(=O)OCC(N2CCCCC2Sc2ccccc2OC)=O)c1 c1(OC)cc(C(N2CCC(NC(=O)Cc3nnc(O)s3)C2)=O)ccc1OC(C)C C(=O)(C1=CC2CCCCCC12)N1CCCC(N(C(c2scnc2Cl)=O)CC)C1 C=C(Cl)CC(C(=O)NCCCC(=O)N(C)C)NC(c1cncnc1C)=O C(=O)(C1=CC(O)C(NC(=O)C=Cc2cnc[nH]2)C1)NC1C(OC)COC1 C(=O)(CCC(C)(C)C)NC1CCC(NC(c2n(COC)ncc2)=O)CC1 CC1(C)CC(NC(c2cc(C3CCC3)n[nH]2)=O)CN1C(C1CC1F)=O N1(C(C2C(CC)C2)=O)CCC(CN(C(=O)COCC(F)(F)F)C)C1 C#Cc1cncc(C(=O)NCC(CNC(=O)C(C)Cn2ccnc2)S(C)(=O)=O)c1 C(=O)(C#CC1CCOC1)N(C1(C)CC(NC(=O)Cn2cnc(=N)[nH]2)C1)C1CC1 N1(C(C2C(C)(C(F)F)C2)=O)CC(NC(=O)COc2ccsn2)CC12CCOCC2 C(=O)(CCC(=O)c1ccc(Cl)cc1)NC(CNC(C1(C(C)C)CCC1)=O)C1CC1 CC1CCC(CNC(C2CCN(c3ccc(Cl)cn3)CC2)=O)N(C(C2(O)CC2)=O)C1 C1(n2ccc(C)n2)CCN(N(C)Cc2csc(Br)n2)CC1 C(=O)(C(CCCCOCC)N(CCC1CCOC1)CC)NCCC N1(C(C2(OC)CCC2)=O)CC(C(=O)NCC2(C)CCCO2)C(C)C1 c1(C(=O)NC(=O)CCCn2cccc2)ccc(CNCCC2CC2C2CC2)nc1 C1(NC(CCSCC(N)=O)=O)CC2(C1)CC(CNC(C1CCCCC1F)=O)C2 N1(CC(=O)NC(CNC(C2(CCC=C)CCCC2)=O)C(C)C)CCCOC1=O C(N=c1[nH]c2ccc(Br)cc2s1)C1CCCC(NC(CCC(C)(C)F)=O)C1 C1(C(=O)NCC2(C(F)(F)F)CCC2)CC(F)CN1Cc1cccnc1Br c1(OCCCC(=O)NC2C(NC(C=CCOC)=O)CCC2)cccc(Br)c1 c1(C(=O)NC2CC(C)N(C(=O)C3CC3)CC2)ccc2c(c1)CCO2 c1(CNC(C(F)OC)=O)cccc2c1CN(C(c1cc(CO)[nH]n1)=O)C2 c1(C(=O)NC2CC(CCNC(C3C(OCC)C3)=O)C2)c(Br)cnn1C(C)C Cc1nc(C(=O)NCCC(O)C(=O)N(CC2CC2)CC2CC2)cc(O)n1 C1(NC(C(CCC)=CCC)=O)CN(C(c2cc(C)c(F)cc2O)=O)CCC1(C)C CC1=NOC(CNC(=O)CCC2CC(NC(=O)C(C)c3cccs3)C2)C1 c1(OC)c(NC2CCCCC2CNC(C2(C)CCCCO2)=O)ncnc1C C(=O)(N=c1ccc(C(=O)OC(C)(C)C)n[nH]1)c1n(C(c2ccccc2)C)ccc1 C1(NC(C(C)OCCCC)=O)C2CC3C(C2)C13C(=O)NCc1ccc(C)cc1F CC1CC(=O)NCC1C(=O)Nc1cccc(C(=O)NCC(=O)Nc2ccns2)c1 N1(C(CC2(CC)CCOCC2)=O)CCCC(CCNC(c2csc(Cl)n2)=O)CC1 O(NC(=O)C(CSCC)NC(c1cccnn1)=O)C(C=C)C C(CCC(=O)N(CC(C)CNC(c1cnn(CCF)c1)=O)C)OCCC CC(C)(O)C(F)(F)C(=O)NCC12CCC(CC1)N2C(C1(C)CCCCO1)=O Cc1csc2c(N3CCC(CCNC(C4CC4(C)C)=O)C3)ncnc12 N1(C(c2n(CC)ccn2)=O)CCN(C(C2CCCC2(C)C)=O)C(CC(F)(F)F)C1 CCC(CC(=O)NC1CN(C(=O)CCSCC(C)C)C(CC)(CC)C1)C(F)F c1(C(=O)NCC2CN(C(C3(CC)CCOC3)=O)C2)csc2cc(OC)ccc12 c1(CN(C)CC2CCCC2)cn(CC(F)CCNC(=O)CNC=O)nn1 N1(C(c2cc(C)c(C)s2)=O)C2CCC1CC(CNC(C1(CF)CCC1)=O)C2 C(=O)(CC(C)(C(F)F)N(C)C)N1CC(CCCCNC(c2c(C)oc(CO)c2)=O)C1 CN1C(=O)CN(CC(=O)N(CCCNC(c2ccnc(C3CC3)c2)=O)C)C1=O c1(COC)noc(CNC(=O)C(C2CC2)NC(c2sncc2C)=O)n1 n1(CC(=O)NCC(CCNC(Cc2cccc(C#N)c2)=O)O)cnc2ccccc12 c1(C(N(C)CC2CCN(C(C(CC=C)CC)=O)C2)=O)ccc2ncccc2n1 c1(C(N(CCC(C(C)(C)C)NC(C2C=CCC2)=O)C)=O)ccc2ccoc2c1 CN=c1nc(N2CCC(C(C)(C)C)C2)[nH]c(=NCc2ccnc(O)c2)[nH]1 c1(CCCCNC(C(C2CN(C(=O)OC(C)(C)C)C2)C)=O)ccc(F)cc1F c1(CSCC)cccc(C(=O)NC2C3CCN(C(C4CCC(CC)CC4)=O)C23)c1 c1(CC(=O)NC(C2OCCN(c3nc(C)nc(O)c3)C2)C)cnc2n1CCCC2 C(=O)(C1CCc2cc(F)ccc21)N1CC2CCN(C(CCS(C)(=O)=O)=O)CC21 C12(C(=O)NCC3(F)CCN(C(Cc4c(C)n(C)cn4)=O)C3)CC1COC2(C)C C(=O)(CCCC(=O)N(C)CCNC(C1CC12CC2(F)F)=O)OC C(CN=c1ccnc(Cl)[nH]1)N(C(=O)C=Cc1ccc2ccccc2c1)C N1(C(CC(C)CNC(=O)CCc2cccn2C)=O)CCNC(=O)CC1 CN1CC(NC(C2CC=CCN2C(c2nocc2Cl)=O)=O)C(C)(C)C1 c1(CC)ccc(C(=O)NC(C)CCNC(c2cc(C(C)CC)no2)=O)cn1 c1(C(N(C)C(c2ccc(Cl)c(N)c2)=O)=O)ccc2c(c1)CCOC2.C12(CC1)CN2 N1(C(=O)Cc2cn[nH]c2)CCN(C(c2c(O)cc(F)cc2F)=O)CC2(CC2)C1 C12(CNC(CSc3cn(C)nc3)=O)CCCC1N(C(=O)CCCF)CCC2 Cc1nc(C(=O)NCCn2cc(CNC(C3(C)CCOCC3)=O)nn2)c(C)n1C N1(C(c2cc(CC)ncn2)=O)CCC(NC(C2CC(C)(F)C2)=O)C(F)C1 c1(C2(C(=O)NCC3C(NC(c4cn(C)nc4)=O)CCC3)CC2)c(F)cccc1Br C(=O)(C(C)(C)CCCNC(=O)CC1CCSCC1)NCC(CC(C)C)O C(=O)(CCCC(C)CC)NC(COCCCNC(c1c(CC)noc1C)=O)(C)C CC1CC(=O)NC(C(=O)NC23CCC(C(=O)NCC(c4nn[nH]n4)C)(CC2)C3)C1 C1(NC(C2N(C(C(C)NC(=O)NC)=O)CC=CC2)=O)CC2CCC(C1)O2 c1(C(=O)NCC2C(Cn3cc(C(C(C)C)O)nn3)C2(F)F)ncn(C)c1C c1(CC(=O)NCC2(NC(C(C)CF)=O)CC2)cc(=O)n(C2CCS(=O)(=O)C2)[nH]1 Cc1ccc(=N)[nH]c1C(=O)NC1CCCCC1NC(c1cc(=O)n(C)o1)=O c1(C(N(CC(C)NC(C2(C(F)F)CC(F)(F)C2)=O)C)=O)cc(S(N)(=O)=O)c[nH]1 C(Cc1ccccc1)(CCNC(C1CC1C(N)=O)=O)NC(COCCC(C)C)=O c1(OC)cc(C)c2c(C(N3CC4CN(c5ncnc(SC)n5)CC4C3)=O)c[nH]c2c1 C(C)(CNC(=O)C(C)CNC(=O)CC(=O)N(C)C)(C(C)C)OC c1(C(=O)NC(CC(C)NC(C2(CCCC)CCCC2)=O)C)cnc(Cl)cn1 c1(C(=O)OCC)coc2cccc(O)c12.N1(C(COCCCOC)=O)CCC2C(N)C12 C1(C(=O)NC2CC(O)(CNC(=O)CCc3cncnc3)C2)CCC2(CC2)C1 CCC(F)C(=O)NCCCN(C(=O)C(C)(C)N1CCCCC1)CC c1(C(C(=O)NC2C(CNC(C3C4(CC(OCC)C4)C3)=O)C2)O)cc(F)cc(F)c1 c1(N(C(c2ccncc2F)C(=O)NCCC)CC)cc(C)cc(C)c1 N1(C(CC(n2c(CC)ncc2)C)=O)CCC(NC(=O)C(=O)NC)C(CO)C1 Cc1cc(C(=O)NC(CNC(C2(O)CC(CF)C2)=O)CO)ccn1 C(=O)(C(C)(CSC)NC(C1COCCO1)=O)NC(c1nn[nH]n1)CC c1(N2CCC(C(F)(F)F)(OC)C2)cc(C)nc(NC(=O)CCOC(C)C)n1 c1(C(N2CCC(CN3CCCOC3=O)C2)=O)ccc(C(C2CC2)O)cc1 c1(C(N2CCCN(CCOC(C)C)CC2)C(=O)NC(CC)C)c[nH]c2ccccc12 Cc1nc(C)c(C(=O)NC2CN(C(C3(C(F)(F)F)CCO3)=O)C2)s1 C1(C)(CNC(COCC(C)C)=O)CN(C(C2CCC(=O)C(C)C2)=O)CCO1 c1(C(=O)NC2CN(C(C(C=C)O)=O)CC(O)C2)cc(Br)c([N+](=O)[O-])s1 c1(OC)c(C(=O)NC(C)CC(C)NC(=O)C(=O)NCCC(N)=O)occc1=O CC1(N(C(=O)CCC2CCN(c3ccccc3)CC2)C2CC2)CCC(=O)N1 c1(OC(COC(C)=O)C(=O)N2CCC(c3cnco3)C2)c(C)cccc1C c1(C2CC(C(=O)NC3CC(C)(NC(c4c(OC)ccs4)=O)C3)C2)ccc(Cl)cc1 N1(c2n(C)c(CCC(C)(C)C)nn2)CC(C#N)(S(C)(=O)=O)C1 c1(OC)ncc(Br)cc1C(c1nnnn1C1CCCC1)NCCC(C)(C)OC C1(CC(=O)N(CC#C)CCO)CN(C(c2cccc(F)c2)=O)CC12CC2 c1(C(=O)NC(CN(C(C(CCCC)O)=O)CC)CC)coc2c1NC(=O)CCC2 N12CCC(C1)CNC(=O)c1csc(n1)C2=O.C(C(=O)OC)SCC.C(C)NC c1(C(=O)NC2C(C)N(C(=O)CCSC(F)(F)F)CC2)cncn(C)c1=O C12(NC(c3c(CC)cccc3)=O)CCC(CN(C(=O)CNC(=O)NC)C1)C2 C1(C(=O)NCC(=CC(=O)NOCc2cn(C3CC3)nn2)C)CC2CCC(C1)C2O Cc1cc(Br)ccc1-c1cn(C2CCCC2C(N2CC=CC2)=O)nn1 C1(CNCCCCN(C)CCO)COCC2(CNC2)O1 CN1C(=O)C(F)CC1C(N1CCC(NC(c2ccc(-c3ccncc3)o2)=O)C1)=O C=C=CC(C)C(=O)NC1CC1NC(=O)C(C)C1CC1 Cc1cncc(CCC(=O)NC2CN(C(C3CC3F)=O)CC2C)c1 C1(NC(C2CN(S(N)(=O)=O)C2)=O)CN(C(=O)C(=O)NCC2CC2)CC2(CC2)C1 CC1CN(C(=O)CCC(C)(C)F)C(C)CN1C(c1ncc(Cl)cc1F)=O n1(CC(=O)NCCC2N(C(c3c(C)sc(O)n3)=O)CCC2)cccc(C)c1=O C1(CC=C)CCCCN1c1nnc(-c2ccccc2Cl)n1CC c1(C(=O)NC2CCC(CNC(C3CSC3)=O)C2)cccc2c(O)nncc12 C1(C)(CCC)CCN(C(=O)C(C)(C)CN(C)C(c2sccc2CO)=O)C1 C12(NC(C(=C(C)C3CC3)F)=O)CCOC(CNC(c3cncc(C#N)c3)=O)(C1)C2 Cc1ccc(F)c(C(=O)NCC2CC(O)CN2C(c2cc3n(n2)CCO3)=O)n1 N1(C(CCCCC#C)=O)C2CCC1CC(NC(c1cc(C(F)F)ncn1)=O)C2 CC(C)C(O)C(C)C(=O)NCC(C(=O)NCc1cn(C2CC2)cn1)C(C)C C1(C(=O)Nc2ccn(C)c2)CCN(C(C2CCN(CC(F)(F)F)C2)=O)CC1(C)C c1(N(CC2ON=C(C(C)C)C2)CC2CC(OC(F)F)C2)ccccc1[N+](=O)[O-] N1(C(C(C(C)NC(C2(CN(C)C)CC2)=O)C)=O)CCC(F)(F)CC1 n1(CC)c(C)ccc(C(N2CC(O)(CN(C(=O)CC(C)P(C)(C)=O)C)C2)=O)c1=O Cc1c(C(=O)NC(c2ccccn2)CNC(C2CCCO2)=O)ccc(F)c1F c1(C(=O)OC)c(C)nn(C)c1N(C(C)COC)C(c1cn(CCSCC)nn1)=O N1(C(C(CC=C)CC(C)C)=O)CCCCC2(CCN(C(=O)C(=O)C(F)(F)F)C2)C1 C=CCC(CNC(=O)C(F)=C(C)C)NC(c1ncoc1-c1cccs1)=O c1(C(=O)NCC23CC(NC(c4n(C(C)C)nnc4)=O)(C2)C3)cc(Cl)ncc1O C1(CC)CN(C(=O)CC2CC(=O)NC2=O)CCN1C(=O)Cn1cc(C(F)F)cn1 N1(C(c2c(OC)ccnc2)=O)CCC=C(C(=O)N2CCNC(=O)CC2C)C1 c1(CC2C3(CCC(=O)NCC3)CCNC2)ccc(S(=O)(=O)CC(F)(F)F)cc1 c1(C(c2nnnn2-c2cccc(F)c2)NCCc2onc(C)n2)n[nH]c(C)c1Cl C1(CCCC)CCC(C(=O)NC2CCC(NC(C3(O)CCC3)=O)CC2)CC1 c1(CC)ccc(C(=O)NC2CN(C(=O)CC3CC3(C)C)CC2(C)C)cc1Br CC1CC(CNC(=O)NCC(=O)N(C)C)N(C(=O)C(C)NC=O)C1 c1(C(N(CCNC(CC(C)C(C)(C)C)=O)C2CC2)=O)cnc2c(cnn2C)c1N c1(C(=O)NC2(C)CCCN(C(CCC(C)C#N)=O)C2)n[nH]c2c1CCSC2 C=CC(C)(CC)C(=O)NC1(CO)CCCN(C(=O)CCOCCCOCC)C1 c1(CC)ocnc1C(=O)NC1CC1CNC(=O)C(F)=CCCF C1(CNCc2c(CC(=O)OC)csc2)COCCN1C(=O)C(C)c1cccs1 C(=O)(C(Cn1cccn1)NC(C1CCCC1O)=O)NC(CCC)C1CCCC1 C(C)(CCC(=O)N(CC(C)C(=O)NC)C)NC(CCOCC)=O C1(NC(C2(OCC)CCOC2)=O)C=CCCC1C(=O)N(CCCC(C)C)C C(=O)(C1=Cc2ccccc2C1)N1CC(F)(C(=O)NCC2(C3CC3)CC2)C1 C1(NC(C2OCC(C)(C)C2)=O)CC12CCN(C(=O)Cc1cccc(C#N)c1)C2 C1(CNC(C(C(C)(C)C)N2CCCC2)=O)C(C2CC2)CCN1C(c1cccn1C)=O c1(OC)ccc2onc(NS(=O)(=O)CC3CCCNC3=O)c2c1 C1(NC(c2c(CC)n(C)nc2)=O)CN(C(c2cc(F)c[nH]2)=O)CC1C1CC1 Fc1cc(Br)ccc1SCCC1=NOCC1 CC1CC(C)(C(N2CCC(CNC(=O)C(O)C3CCCC3)C(C)C2)=O)CC(C)O1 C(=O)(C1CCCc2ncccc21)NCC(C)NC(Cn1ncc(C#C)c1)=O c1(CN(C(C)C)C(=O)NCCC(c2ccccc2)N(C)C)ccc(Cl)cc1 C(=O)(C(CC(N)=O)NC(=O)CC1(O)CCCCC1)NC(CC#C)CC#C c1(NC(CNCc2cccc(C)c2)C(C)C)scc2c1CCCC2 CCC(CC(=O)NCC1(C)CCCN(C(=O)COCCCOC)C1)C(F)F N1(C(CC(CCC)CC)=O)CC2(C)CN(C(=O)C(C3CCC(=O)N3)C)CC2(C)C1 C12(C(N(CC(F)C(=O)NC)CC#C)=O)CC1CN(C(=O)COc1ccn(C)n1)C2 c1(-c2cc(C(=O)NCc3cccnc3Br)c(F)nc2)cnc2c(F)cccc2c1 [N-]=[N+]=NC1CCC(C2CC2C(=O)NCc2ccc(OC(F)F)cc2)C1 c1(C(N(CC(C)NC(C(COC)N(C)C)=O)C)=O)c(Br)ccc2n[nH]cc12 C(=O)(CC1NC(=O)c2ccccc21)NC1(CC=C)CN(C(c2occc2Br)=O)C1 S(=O)(=O)(c1cccc(Cl)c1F)NC1CN(C(c2ccnc(OC)c2C)=O)CC1O C1(NC(c2n(-c3cccc(OC)c3)nnn2)C2CC2)CCC2CC(F)(F)CC2C1 C1(CC(=O)N(C(C)(C)CN2CCc3ccccc32)CCO)CCC2(CC(C(=O)O)C2)O1 N1(C(C(N2CC(CCNC(C(CC)=CC)=O)C2)=O)C)CCN(C)CC1 C1(C(N2CCCC(F)(CNC(C(C)C3CCOC3)=O)C2)=O)CCc2ccnn2C1 c1(NC(C(=O)NC2(CC)C(OC)C(C)C2OC)=O)ccc(OC)cc1[N+](=O)[O-] CC(C)C(C(=O)N1CC(NC(C2CN(C(N)=O)C2)=O)C(O)C1)c1cccc(Cl)c1 C1(CCCNC(CC)C(O)c2ccccc2)CCCNC1=O C(C)(C)(CC(=O)NCc1cnn[nH]1)NC(COCCC=C)=O CC(=O)C(C)CC(C)C(=O)N1CC(O)CCC1C(=O)NCc1noc(C)n1 CCCCC(C)CCC(=O)NCC1CCC(C(=O)NOCC(F)F)C1 C1(NC(CCC=C)=O)CC2CCC(C1)N2C(=O)COc1ccc(Cl)nc1 c1(C(N2C(C)(CNC(c3cnc(C(C)C)s3)=O)CCC2)=O)csc2cncn12 C(=O)(CC(C)(C)C)N1CC(C(C)NC(C(C)c2ncco2)=O)C1 c1(CC(C)N(CCN2CCN(C(=O)NC)CC2)CC)noc2cc(Cl)ccc12 CC(C)(C(=O)NC1C2CCC1N(C(C1(CC3CC3)CCC1)=O)C2)S(C)(=O)=O C(=O)(C1=NOC(C)(C)C1)NC(CCOC)CNC(=O)C(c1ccccc1)OCC N1(CCC(N2C(CNC(CN3CC(C)(OC)C3)=O)C=CC2)=O)CCNC(=O)C1 C=Cc1ccc(C(N2CC(NC(c3cc(Br)cnc3O)=O)C(F)(F)C2)=O)cc1 C(CC1CC1)(C(=O)OCC)N(C(=O)NCC(=O)N(CCOCC#C)C1CC1)C C1(C(=O)NCCCC(C)NC(Cn2c(C)nnn2)=O)CCC(CO)CC1 N1(C(C2N(C(=O)NC)CCC2)=O)CC2CC(C1)CN(C(C1CC(OC)C1)=O)C2 c1(C(=O)NCCN(C(Cc2c(C)nsc2)=O)C2CC2)cn(CC(F)F)nc1C C1(C(N2C(CCNC(c3cc(CC)n(C)n3)=O)CSCC2)=O)CCCCC12CC2 N1(C(C2C(C(C)=O)C2)=O)CC2CC(C1)N2C(=O)CC1(N(C)C)CC1 C1(CC(=O)NCc2cc(COC)no2)CCCCC1NC(C1CC1F)=O C(=O)(CC(C(C)(C)C)NC(=O)Cc1cncs1)NC(C1CCOC1)C C(C(CC(=O)NCC1CCN(C(C)C)C1)OC)NC(CC1CC(=C)C1)=O c1(C(=O)NC2CCC3CCN(C(C(CC)CC)=O)C32)ccc2c(c1)C(=O)C(=O)N2 c1(-c2c(C)occ2)nc(CC(O)CF)n(C(C)C2CC2)n1 c1(C(N(C(C)CCNC(c2ccc(C3CC3)o2)=O)C)=O)ccc(S(C)=O)cc1 C(C(C)(C)C(=O)N1CCOC(CCNC(=O)C(C2CCCOC2)OC)C1)OCC c1(OC)cc(C)c(C(=O)Nc2ccsc2C(=O)Nc2ccc(O)cc2C)cn1 N1(C(c2c(C)con2)=O)CC2(CC(C(N3CCCC3(C)CC(C)C)=O)CO2)C1 c1(CC(=O)NCCNC(C(CC)(C)F)=O)cc(F)cc2c1OCOC2 C1(C(C)(C)C)CC(C(=O)NCC2CCCCC2NC(=O)COC2CCCC2)=NO1 c1(CN(C(=O)NC(C#C)C2CC2)CC)ccc(SC)o1.C(=O)(C(C1CC1)C1CC1)N C(=O)(C(C)(C)CO)N1C(NC(CN(c2ccccc2)CC)=O)C(C(F)(F)F)C1 c1(NC(C2CC(=C3CCC3)C2)=O)nccc(CN2CC(N3CC=CC3)C2)n1 c1(C(N2CC(c3cccc(Cl)c3)C(O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 C1(NC(C2CCCC2)=O)CCN(C(C2CCCCO2)=O)CCC1CO c1(C(=O)NCC2CCCN(C(C3(NC(C)=O)CCCC3)=O)C2)ccc(C#N)n1C c1(N2C(=O)C2)ccc([N+](=O)[O-])cc1.C1(c2cn(C(C)C)nn2)C(C)CCN1C1CC1 CCCC(CNC(c1cccc(CNC(=O)C(C)CC(C)C)n1)=O)CCC c1(CCCC)ccc(C=CC(=O)NC2CC2N(C(=O)C=C(C)c2ccsc2)CC)o1 C(=O)(C(N=[N+]=[N-])C(C)C)N(CCC(=O)Nc1cc(C)c(C)nc1)CCO CCC(C(=O)NC1CCCC1CNC(c1cc(CN(C)C)c[nH]1)=O)N(C)C c1(CCC(N2CC(COC)C3(C2)CC3)=O)ccnc2ccccc12 N1(C(C23CC2CN(C(=O)C(Cl)Cl)C3)=O)CCC2(CCOC2)CC1 c1(C(N2CCC(F)(C(=O)NC3CCCC(O)C3)C2)=O)ccc(O)cn1 c1(C(C)(C)NC(=O)CSC2CCc3[nH]nc(C(F)(F)F)c3C2)nnc2n1CCCC2 C1(C(=O)NCC2(C)CCN(C(C(F)=CC)=O)C2)CCC2C(=O)NCC(=O)N2C1 C1(CCNC(C2C(OCC)C2)=O)CCN(C(=O)CC(=O)Nc2ccccc2)CC1 c1(OC)ccc(C(F)(F)C(=O)NC(C)CC(C)NC(=O)CCCCC2CC2)nc1 C1(OC)COCC1NC(=O)C(F)C1CC(C(=O)OC(C)(C)C)C1 c1(CCCC(=O)NCC2CCN2C(C2CCS(=O)(=O)N2)=O)nc2ccccc2o1 N1(C(COc2cn(C)nc2)=O)CCCCC1C(=O)NC(C1CCCO1)(C)C N1(CCC=CCCC)CCC(N(C(=O)CC(C)n2ccc(C)n2)CC)CC1 N1(C(C(C)CBr)=O)CCC2(CCCC2C(N2CCCOC(CO)C2)=O)C1 N1(C(c2cnn(C)c2C#N)=O)CC(C)(C(N2CC(CO)C(O)C2)=O)CC1(C)C n1(CCOCC)nnnc1C1(NCC2(C)CC2(Cl)Cl)CC(CF)C1 Cc1ccc(C(=O)NCC2CN(C(=O)C(C)C3CCCO3)CCC2C)c(F)c1F c1(C2(CNC(C3CCCN(C(c4cc(C)on4)=O)C3)=O)CC2)cc(F)ccc1Cl C1(C(N(C2CCC2)CC)=O)CC=CC(NC(c2cn(C3CC3)cn2)=O)C1 Cc1cc2c[nH]nc2cc1C(=O)NCC(O)CN(C(=O)CCC1CC1(Cl)Cl)C n1(CC(N2CCCCC(NC(C(C3CCCC3)OC)=O)C2)=O)cc(F)ccc1=O c1(C(=O)NC2CCC(CCNC(=O)CSc3cccs3)C2)cc2ccccc2[nH]1 c1(C(C(=O)NCCN(C(c2c(C)cc[nH]2)=O)C2CC2)(F)F)ccc(Br)nc1 c1(C(=O)NCC2CCCO2)cc2c(s1)CCN(Cc1ccc([N+](=O)[O-])o1)C2 C1(NC(c2ccn(COC)n2)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(C)O N1(C(c2cnnc(C)c2C)=O)CCC2CN(C(=O)C3CCc4nccn43)CC2C1 C12(C(N3CC(CNC(C4CCCOC4)=O)OCC3)=O)CC(CO)(C1)OC21CCC1 c1(C(=O)NCC(CNC(COCCOCC)=O)O)c(Cl)ccc(O)c1N C1(C(=O)Nc2cccnc2CO)CC(F)(F)CN1C(=O)CC1(O)CCC1 c1(C(N)=O)cncc(C(=O)NC2CC(CCNC(c3ncncc3Br)=O)C2)c1 c1(OC)nccc(C)c1CNC(=O)NCCc1ccncc1F c1(NC(C2N(C(c3c(CCC)nco3)=O)CC(O)C2)=O)ccc2c(c1)COC2 Cc1cc(NC2CCN3CCC2C3)ncc1S(=O)(=O)NCc1ccc(CO)o1 Cc1ccnn1CC(=O)NCCn1cnc(C(=O)NC(C)CO)c1 Cc1oc(CO)cc1C(N1CCC(CF)(NC(=O)C2CC2)C1)=O.c1(S)ccncc1F N1(C(Cc2cc(C)cc(C)c2)=O)CCN(C(=O)C2=CCCCC2)CCC1C N1(C(=O)NCc2cnc(CC)s2)CCC(O)(COC2CCOC2)C1 C(=O)(CCCn1ccc(C(=O)N)n1)NCCN(C(C1(NC(N)=O)CC1)=O)C.C1CC1 N1(C(C2N(C(c3n(OC)cnc3C)=O)CC2)=O)CCC2(CNC(=O)N2)C1 CC1CN(C(c2cccc(=O)n2C)=O)CC(CCNC(c2sccc2CO)=O)O1 N1(C(c2cccc3ccoc23)C(=O)NC(C)C)CCC2OCCCC2C1 c1(C(N(C)CC2N(C(CC3C(C)=NNC3=O)=O)CCC2)=O)c(O)nc(=N)[nH]c1C C1(NC(COc2c(C)noc2)=O)CC(C)CCC1Cc1ccccc1 c1(C(N2CCOCC2Cc2cn(CC(F)(F)CO)nn2)=O)ccc2scnc2c1 n1(CCOC)cc(NC(=O)C(O)CN2CCOCC2)cn1.C12(CCC1)C(=O)NC2 c1(CN(CC(F)(F)F)CC(N2CCCC(CS(C)(=O)=O)C2)=O)ccc(C#N)cc1 CCC(C)(COC)C(=O)NCCCCC(=O)Nc1cc(C)ccc1CO Cc1cc(CNC(=O)COC2CCN(C(c3ncccc3N)=O)C2)sc1C C1(C)(C(=O)NCCCC(C)NC(C2CC(F)C2)=O)CCCOC1 C1(CCCC)CN(C(c2cn3ccsc3n2)=O)CCN1C(=O)Cc1ccns1 C1(C)(C(=O)NC2CCCN(CCC)C2)CCCN(C(=O)C=Cc2ccc[nH]2)C1 c1(NC(C(n2nnnc2-c2cc(Cl)ccc2Cl)CC)=O)cc(F)c(Br)cc1C n1(CC)ncc2cc(C(=O)N(C3CN(C(=O)CC4CCCC4O)C3)C)c(C)nc12 C(=O)(C(C)(C)CCC)NCC(CNC(c1cnc(CCC)s1)=O)O c1(CC)ncc(C(=O)N(CC(O)CNC(c2nocc2C(C)C)=O)C)s1 N1(C(CN2C(C)CCC2)=O)CCC2(CC1)CN(C(=O)C(CO)C(C)(C)C)CCO2 C1(C(=O)NOCCC(C)(C)C)(OC)CCC(C)(C)C1.c12c[nH]nc1NC2=O C=CC1CN(C(=O)CCC2(C)CCC(=O)N2)CC1NC(c1cc(COC)on1)=O N1(C(Cc2cc(C)nn2C)=O)CC2CC(NC(C3(N(C)C)CCC3)=O)C(C2)C1 c1(C(N2CC(N(C(c3c(COC)noc3)=O)C)C(F)C2)=O)c([N+](=O)[O-])cnn1C S(=O)(=O)(c1cccnc1NCC1(CC2CCC2)CC1)N1CCN(CC(C)O)CC1 CC(C)CC(O)C(C)C(=O)N1CCSCC1C(=O)N(C)Cc1ncnn1C C1(N(C)C(c2ncoc2C(F)(F)F)=O)CCC(NC(=O)CCc2nncn2C)C1 c1(C(=O)NC2CCN(C(CCC(=C)C)=O)C2)c2c(nn1C)CCOC2 c1(C(=O)NCC2N(C(C3CC(C(=O)OC)C3)=O)CCCC2)ncc(Cl)cc1F C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NC(CCC(=O)NCCCP(C)(C)=O)=O c1(C(=O)NC2C(NC(c3ccc(Cl)s3)=O)C2)sccc1Cl CC(C)C(C(=O)NC1CC(C(c2ccccc2)=O)C1)NC(C1CCCOC1)=O C1(C)(C(=O)NCC2(CO)CN(C(CCOCCCOCC)=O)C2)CCN(C)CC1 C1(C)(C(=O)NCC(COCC)O)CCN(C(C2CCC(=O)C2)=O)CC1 c1(C(C=C)N(C)C)nc(C2CCOC2)nn1CCC=C c1(C(=O)NC2C(NC(CSCC)=O)C2)cc(NCc2ccccc2OC)cc(N)c1 C(=O)(C(C(C)O)NC(=O)NC1CC1c1nc(-c2cc(Cl)cs2)no1)OC N1(CCC(=O)NCC(CNC(c2cscc2C(N)=O)=O)OC)C(=O)CCC1=O c1(C(=O)N)ncc(C)cc1C.C1(OC)CCCC(CNC(C2(CO)CC(C)(C)C2)=O)C1 C(CN=C(NC(C)C1CC1)NC1CSC1(C)C)c1ccc(SC)cc1 C#CC1(NC(C2CCC3(CC3)N2C(C2C3CCC(F)C23)=O)=O)CCCCCC1 O=C(C1=NN2CCCN=C2N1)NC12CC1CN(C(=O)C(F)CC1CC1)C2 CC1(C)Cc2cc(C(=O)NCC3C4CN(C(C5CCC(=O)O5)=O)CC34)ccc2O1 c1(C(C)=O)cc(C(=O)NC(C)CCNC(c2c(OC)cccc2O)=O)ccc1C c1(C(N2CCC(CC(N3C(C#N)C4CC4C3)=O)C2)=O)cc2n[nH]cc2cc1Cl C=C(C)C(C)(C)C(=O)NCC1(CNC(=O)Cc2cc(Cl)sc2Cl)CCCC1 C1(O)(C(C)NC(=O)CCOc2ccc(Cl)cc2)CCN(C(=O)C(=O)N(C)C)CC1 C1(NCc2c(C(N(C(=O)NC)CC)=O)ccs2)CN(C)CC1C(F)(F)F N1(C(C(=O)NCCC#N)c2cn[nH]c2)CCC2(CCC2)C1 Cc1cc(=NC(=O)N2CCC(C=CC(=O)Nc3cnsc3)CC2)[nH]n1C(C)C C(=O)(C1=C(C)CC1)NC1(C(N2CC(C(=O)NCCCCC)C2)=O)CN(C(C)=O)C1 C1(C(=O)NC2COCCN(C(=O)C(C3CC3)C3CC3)C2)CC2CCCCC2C1 N1(C(CN(C)C)=O)C2CCC1CC(N(C)C(C1C(C)(C)C1(C)C)=O)C2 Cc1cn2c(n1)CC(C(=O)N(C)CCOCCNC(C1(F)CCOC1C)=O)C2 C(=O)(C1=CC2CCC(C1)C2)N1C(C)(CC(=O)NCC(CC)CO)CC1 O=C(C1=COCC1)NCC1CN(C(c2occc2Cl)=O)C1 N1(C(C(C(C(C)C)OC)O)=O)CCNc2cccc(C(F)(F)F)c21 c1(C(N(CC(CC)NC(C2CCCC2CN(C)C)=O)C)=O)ccnc(CO)c1 C1(CNC(c2ccc(C(C)=O)[nH]2)=O)CC2CCCC2N1C(=O)C#CC1CCC1 C1(C(N2C(COC)CCC2)=O)CN(C(C2CC3(CSC3)C2)=O)CC1(F)F S(=O)(=O)(c1ccccn1)NCC1CCN(C(c2c(OC)cccn2)=O)CC1(F)F c1(CN)cccc2[nH]ncc12.N12CC(C1)NC(=O)NCC2=O.CN c1(C(C)NC(C(COCC)n2cc(COC)nn2)=O)cc2cccnc2s1 CC1(C(=O)NC2CCCC2CNC(C2(C)CS(=O)(=O)C2)=O)CCSCC1 N1(C(COCCOC)=O)CC(CNC(C2CC(F)(CO)C2)=O)CCC1C C1(N(C(=O)CCOCCCN(C)C)CCC)CCN(C(=O)C(C)SC(F)(F)F)C1 c1(-c2cn(CC3C(N4C(C)CCCC4)CCCC3)nn2)c(Cl)cnc(Cl)c1F CCC(CC)C(=O)N1CCC(CNC(C2CC2C(=O)OC(C)(C)C)=O)C1 N1(C(c2ccc(N)c(F)c2)=O)CCCN(C(C2(C)CSC2)=O)CCC1 C1(C(N(CCNC(=O)C(C)c2ccco2)CC)=O)CC12CCS(=O)(=O)CC2 C1(NC(C=CC)=O)CCCN(C(=O)CC2C(=O)ON=C2C)C1C CCC(C(=O)NC1CCCC1NC(C1CCC(=O)N1)=O)OC C1(CC(C(=O)NC)N(C2CC(F)(F)C2)C)COC(C)(C)C1 c1(C(=O)NC(CC2CN(C(COC(CC)C)=O)C2)C)cnc2n1CCS2 c1(C(C)NC(=O)NC2C(CC(=O)OC)CCC2)ccc(OCF)cc1 C12(NC(C3(CNC(c4cc(C(C)C)nn4C)=O)CC3)=O)CCC(C1)OC2C CC(C)CC(=O)NCC1CC1CC(=O)NC(C)COC(F)(F)F c1(OC)ccc(-c2cn(CCC(=O)Nc3ccco3)nn2)cc1.C1(C)C(=O)N1 N1(C(C2C(C)=CCS2)=O)CCCCC2(CCN(C(c3cc(Cl)ccn3)=O)C2)C1 C(C(O)CC(=O)NCC1(CNC(=O)CC(C)(C)C)CC1(F)F)N(C)C.C1CO1 C(=O)(C1=CC2(CCOCC2)C1)N1CC(N(C)C(=O)C2CC2)C(F)C1 c1(C(N2CC3C(NC(c4c(C)nc(C)s4)=O)(CC3)C2)=O)cnc([N+](=O)[O-])n1C C=CC1OCCC1N=c1[nH]c(=NCCC2OCCC2(C)C)[nH]c2cc(C)ccc12 c1(C(N2CCC(N(C(C3CC(C(=O)OC)C3)=O)CC)C2)=O)cc2c(s1)CCSC2 C1(CC)C(C(N2CC(O)(CO)C2)=O)CCCN1C(=O)Cc1ccnc(O)c1 c1(-c2nnc(N3Cc4c(nc(C)s4)C3)n2CC2CC2)cc(Cl)cc(S(C)(=O)=O)c1 N1(C(C(CCC)OC)=O)CC(NC(c2cn(CC)nn2)=O)C(S(C)(=O)=O)C1 CC(C)C(O)CC(=O)N1CCC(C(C)NC(=O)COCC(N)=O)C1 N1(C(C2N(C)C(=O)CC2)=O)CC2(CC(CC(N3CCCNC(=O)C3)=O)C2)C1 CC1CCC(NC(C2CCCC2C2CC2)=O)CN1C(=O)Cn1cccn1 c1(C(=O)NCC(CC)(C)OC)cc(C)c2[nH]c(=N)sc2c1 NC1CC=CCC1C(=O)NCc1nc(Cc2ccc(F)cc2)cs1 c1(C(=O)NC23CC(CNC(c4c(SC)cnn4C)=O)(C2)C3)cc2ccccn2c1 c1(NC(N2CCCC(C(=O)Nc3ccccc3)C2)=O)ccc(Br)c2ncccc12 Cc1nc(CC(=O)NCC(C)(C2CC2)NC(=O)C(O)C2CCCC2)c(C)s1 Cc1cc(C(=O)NC(CNC(C2(C)CCCO2)=O)C2CC2)c(O)c(C)n1 C1(NC(C2(C(C)(C)O)CC2)=O)CCCC(C(=O)NCCCCC2CCCC2)C1 N1(c2cc(OC)nc(OC)n2)CCC(NC(=O)CC2CCCCN2C)C12CCC2 N1(C(C2CCN(C)C2)=O)CC2OCCN(C(=O)CC3(C(F)F)CC3)C2C1 CCC(C)(C)CCCC(=O)N1CC(O)(C2CCCN2C(=O)CC2CC23CC3)C1 CC(C)CC(CNC(C12CC(C)(CO1)C2)=O)NC(=O)C(C)SC(F)(F)F S(=O)(=O)(C1CC1c1ccccc1NCc1ccccn1)NCCCOC(C)C N1(C(COCC(C)(C)C)=O)CCC2CCC(NC(=O)CCCCF)C1C2 c1(OC)ncnc(C(=O)NC2CN(C(C3CCC(=O)O3)=O)CC2C)c1F C#CC1CN(C(C2CCC(C)(C)CC2)=O)CCN1C(C1CC(n2ccnc2)C1)=O C1(N(C(CC(C)OC)=O)C)CCN(CCC2CCCC(C)C2)CC1 C1(OC)(CNC(=O)C(CC)SC)CCN(C(=O)C(F)(F)c2nccn2C)C1 CCCCCCCC(=O)N(C(C)C(=O)N(C1CC(CC)C1)C)C N1(C(C(=Cc2ncn(C)c2)F)=O)CC2(CC(NC(C3COCC3(C)C)=O)CO2)C1 c1(C(C)N(C(C(N2C(CC)CC(OC)C2)=O)=O)C)cc(F)ccc1C C1(C(C)C)C(C(N2CC(O)C(O)C2)=O)CCN1C(c1ccccc1F)=O c1(N2CC3(C)CN(C(CSCCC)=O)CC3(C)C2)ncnc2c(Cl)cc(Cl)cc12 N1(C(C(COC)NC(=O)NC)=O)CC2CC1CN(C(c1cnc[nH]1)=O)C2 C12(C(N3CCC(C)(NC(CCNC(=O)OC)=O)C3)=O)CCC(C(F)F)(CC1)C2 C1(C(N2CCC(C(=O)OC)O2)=O)CCc2cnn(C)c2C1 c1(C(=O)NCCN(C(c2noc(C3CC3)c2C)=O)CC)cc(C)cc2ccoc12 N1(C(C23CC(NC(C(COCC)C)=O)(C2)C3)=O)CC2(COC(C)C2)C1 CC1CN(C(=O)CSC2CC2c2ccccc2)CC1(C)C(=O)O N1(C(C2(C3(C)CC3)CC2)=O)CCC(C(=O)N2CCCC2CCCO)=C(F)C1 N1(C(C(C)SCC)=O)CC2(C1)CN(C(=O)CC1=CCCCC1)CCO2 c1(OCc2nc(-c3ncn(CC(=O)OC)n3)on2)ccc(Cl)cc1Cl C1(C(=O)NC2CC(C)(CNC(CCOCC#C)=O)C2)CCc2nnc(C)n2C1 c1(C(=O)NCC(C(C)(C)C)NC(C(C)C2CCC2)=O)cccc([N+](=O)[O-])c1 CCC(C)C(O)C(C)C(=O)NC(CC(=O)NC1CCN(CC)CC1)C(C)C N1(C(CC2N(C)CCCC2)=O)CCC2(CC1)CN(C(=O)Cn1cccc1)CCO2 C1(NC(c2n(CC)c(O)nc2)=O)CCC(C)N(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 c1(CC(=O)NC2(CCCCNC(C(C)N(C)C)=O)CC2)cc2ccccc2s1 N1(C(CCCC#N)=O)CC(C2CCCN(C(C3CCC(C(N)=O)O3)=O)C2)C1 N1(C(Cn2c(C)ccn2)=O)CCC(N(C(C2CCCCO2)=O)C(C)C)CC1 CCCC(C)C(C)(c1nnnn1CCCSC)NCCCCCC(C)C N1(C(c2ccc(OC)s2)=O)CC2CCC(CNC(c3ccnnc3)=O)C2C1 N1(C(C=C(C)Cl)=O)CC2CCCC(CNC(=O)C=C(C)c3ccco3)C2C1 N1(C(c2c(N)cc(F)c(Cl)c2)=O)CC2CC(C1)CN(C(c1ccnc(S)c1)=O)C2 C(=O)(C(C(C)C)NC(=O)CCSCC(N)=O)NCCC(C)(C)OC C(=O)(C(CC(F)F)c1ccccc1)NC(CCN(C(c1nccc(C)n1)=O)C)C CC(C)(C)C(C(=O)N1CC2(CC(NC(C3(CO)CCC3)=O)C2)C1)C1CCC1 C1(NC(CNC(c2c(C)occ2)=O)=O)CCCC(NC(c2nc(O)sc2C)=O)C1 C=CCC(CC(C)C)C(=O)NCC1CCN(C(c2cccc(N)n2)=O)CC1(F)F Cc1nn(C)c(C)c1C(N1CC2(CCC2NC(C2CCCN2C=O)=O)C1)=O C=CCCCC(C(=O)NC1COCC1F)NC(C1CC12CCCC2)=O S(=O)(=O)(c1ccc(F)c(F)c1F)NC1CCC(C(=O)NC2CC2(F)F)CC1 c1(-n2c(CC(F)(F)CC)nc(C(CCC)C)n2)c(C)nc(C(C)CC)nc1C C(=O)(C(C)C(C)S(C)(=O)=O)N1CC(C(C)NC(c2cn3cccnc3n2)=O)C1 C1(C)(NC(CNC(CCCC)=O)=O)CCCC1C(=O)NCC(c1ccsc1)C N1(C(c2c(C)nsc2)=O)CCOC(C(C)NC(=O)CC23CCC(CC2)C3)C1 C1(C(=O)NCCc2ccccc2O)CCCCCN1C(=O)CC1CCC1 C1(NC(c2cnc(C)[nH]2)=O)CCCCC12CCCN(C(=O)CCOC(C)C)C2 c1(C(O)CNC(=S)Nc2ccccc2F)ccccc1[N+](=O)[O-] c1(CC(=O)NCCC(=C)CNC(=O)C=Cc2cncn2C)c(C)cccc1Br C1(C(=O)NC(C(=O)NCC2CN(CC)C(=O)O2)c2ccoc2)CC1C1(C)COC1 c1(C(=O)N(CCO)CCc2ccncc2)ccc(Br)o1.n12cc(nn1)SCCC2 CCCC(Cc1ccccc1)C(=O)NCCN(C(c1cc(C)c(O)nn1)=O)CC C1(C(N(CCC(=O)NC(C)C(C)(C)C)C)=O)CN2CCC1CC2 c1(N(C(C)C2CC2)C(=O)NCCCN2CCOC2=O)c(F)cccc1F Cc1ccc([N+](=O)[O-])c(NCC(C2CCCC2)NC(=O)Cn2cncn2)c1 c1(OCC(=O)N(CC(CC)NC(c2cnc(C)[nH]c2=N)=O)C)ccc(F)cc1F c1(C(=O)NC(CNC(CCCSC)=O)C(C)C(C)C)cc2nc[nH]c2cc1N C=CC(C)(C)CNC(=O)C(C1CCC1)NC(c1sccc1OC)=O c1(CC(=O)N(CC(C)NC(CCC=CCC=C)=O)C)ccc(C#N)cc1F C(=O)(C(C)C1=CCCC1)NC(CC=C)CNC(=O)C1=CCCCC1 c1(C(N(CCNC(=O)CC2(C)CCCO2)CC)=O)n[nH]c2c1CN(C)CC2 N1(C(c2ncn(CC)c2)=O)CCN(C(c2ccco2)=O)C(C(C)C)C1 CCCCCCCC(=O)NC(C1(O)CCN(C(c2ccc(C)cc2Cl)=O)C1)C c1(NC(C(N2CCC(C3NCC3(C)C)CC2)C)=O)c[nH]c2ccc(Br)cc12 c1(C(=O)NCCCN(C(c2c(SC)csc2)=O)C)ncccc1C c1(CC(C(=O)OCC)NC(C2(COC)CCCN2)=O)cc(Cl)ncc1F N1(C(C(C)OCC=C)=O)CCCC(C(C)CNC(C2CC(=C(F)F)C2)=O)C1 CCC(C(O)C(F)(F)F)NC(=O)C(=O)NC(c1cccc(Br)c1)c1nc(C)no1 C(C)(C)(CCCCNC(=O)COCC1CC1)NC(C(C)n1cccc1)=O c1(OCC)ccc2nc(N3CCCCC3CNC(C3(C)C=CCC3)=O)sc2c1 C1(C(N2CC(NC(C3(CF)CC3)=O)C2)=O)CC2CCCCC2O1 C12(C(=O)NC3CC4CN(C(C(CCCC)O)=O)C3C4)CCCCC1CCCC2 C1(NC(C2N(C(COCCSC)=O)CC=CC2)=O)CC=C(C(C)C)CC1 N1(C(CC2C(=O)NC2)=O)CCCCC1C1CC1 N1(C(C(C)(N(C(c2c(CC)occ2)=O)C)C2CC2)=O)CCC(CC)(CO)C1 N1(C(C2C(OCC)CCC2)=O)CCCC(C2CC2NC(c2ncc(Cl)n2C)=O)C1 Cc1cn2cc(C(=O)N(C(C)CCNC(C3COC3)=O)C)nc2s1 O=C(C1=CC2C=CC(C1)C2)NC1(CNC(c2cncc(O)c2)=O)CCOC1 c1(CCC(=O)NC(CN(C(c2n(CC)ccc2)=O)C)C)c(F)cccc1Cl c1(CCNC(=O)NCC2(N=[N+]=[N-])CC2)nnc2n1CCCCC2 Cc1nc(CC2CC=CC2)sc1C(=O)N(C1C2CN(C(c3cnn[nH]3)=O)CC12)C N1(C(CCC2C(C)=NOC2=O)=O)CC2(CCCCN(C(=O)CC3=CCCC3)C2)C1 N1(C(C(C)CC2CC2)=O)CC(NC(c2ccc(-c3ncc[nH]3)cc2)=O)C(CO)C1 C1(COC)(NC(=O)CCN(C)CCO)CCN(C(C2(C(C)C)CC2)=O)CC1 C(C)(C)(CCN=c1cc(C(C)(C)C)nc(Cl)[nH]1)NC(C(C)Cc1ccco1)=O N1(C(CCCC#CC)=O)CC2ON=C(CNC(=O)CCn3ccc(C)n3)C2C1 N1(C(CC(n2c(CC)ncc2)C)=O)CCCN(CCNC(C2(SC)CC2)=O)CC1 c1(C(C(=O)NC(CC)C)N(C(C)C(=O)NC2CC2)C)ncc(COC)s1 c1(C(C(=O)NCC(CNC(c2ccc(C(C)C)s2)=O)C)C)ccc(F)cc1 NS(=O)(=O)c1cc(C(=O)NCC2C3CCC23)c(Cl)c(F)c1 C1(C(=O)NCC2CC(CNC(c3ccc(O)cc3F)=O)OC2)CC2C=CC1CC2 C1(C(C)NC(CN(C)CC)=O)CN(C(=O)C(C)C(C)c2ccc(F)cc2)CCO1 CC1(C)C2CCC(C(=O)NCC(O)CNC(C3(F)C(C)(C)C3(C)C)=O)C1C2 C1(CC)CC(C)CN(C(C2(C(C)C)CCCN2C(c2ccn(CCF)n2)=O)=O)C1 Cc1ccc(CC(=O)NCC(CC(C)C)NC(=O)C(c2ccccc2)F)c(C)c1 Cn1nc2c(c1NC(C13CC1CN(Cc1ncccc1[N+](=O)[O-])C3)=O)CCCC2 C#Cc1cccc(C(=O)NCC2CC(F)(CNC(C3(F)CCOC3C)=O)C2)c1Cl C#CCC(C)(CNC(c1ncoc1CNC(=O)CC1CCSCC1)=O)CO Cc1ccc2c(C(=O)NNC(C3(C)CCCS3(=O)=O)=O)[nH]nc2n1 Cc1cc(C(=O)NC2CCC2C(=O)NCCOCCCO)cs1 CC1(C)CC(CNC(=O)Cn2cc(CO)nn2)CN1C(=O)C1=C(Cl)CCC1 CCC(C)C(C(=O)NCC1CCN(C(=O)c2csc(COC)n2)O1)N(C)C C(=O)(CC(C)CC(=O)N(CC(C)NC(c1ccc(N2CCCC2)cc1)=O)C)OC C1(O)(CNC(c2c(C)sc(O)n2)=O)CCCN(C(=O)CC2(O)COC(C)(C)C2)C1 N1(CCOC)CCCC(CN(c2ccccc2C)C(c2cn(C)nn2)=O)C1 N1(C(c2ccc3cncn3c2)=O)CCC2(CCN(c3ncnc(O)c3Br)C2)C1 CC1(C)CCCN(C(C2CCCCN2C(c2cncn2-c2ccccc2)=O)=O)C1 c1(C(CC(C)NC(C2CCC3(CC3)C2)=O)NC(=O)CC(C)(C)C)ccc(F)c(F)c1 c1(C(C(=O)NC(C2CCCO2)COC)C)cncn1C c1(C(N2CC(CN3CCN(C(CCC=C)=O)CC3)C2)=O)cc(=O)n(CC)n1C N1(C(C2=CC(C)(CC)C2)=O)CC2(CCN(C(=O)CC3CC(C(C)(C)C)C3)C2)C1 C1(C(N2CCC(C(C)NC(=O)C(F)CC(C)C)CC2)=O)(OC)CCCCCCC1 C12(C(=O)NC3C(C)(C)CN(c4nc(Cl)c(C#N)s4)C3)CC3CC(C1)C(=O)C(C3)C2 C1(CNC(C(C(=O)OC)C)=O)CN(C(c2cc(C(C)C)nn2C)=O)C(C)(C)C1 N1(C(C2(CC)CCC2)=O)CCOC2(CCN(C(C3CCCCS3)=O)C2)C1 n1(CCCC(N2C(C)CC(NC(CCC=C(C)C)=O)C2)=O)nc([N+](=O)[O-])cc1C C1(CC)CN(C(c2cnc(C)cc2C)=O)CCN1Cc1cccc(C(F)F)n1 c1(CCC)cc(C(=O)NC(C)CC(C)NC(c2ccnc(N(C)C)c2)=O)n(C)n1 C(C(CC(C)C)C(=O)NC(C)C(=O)OC)NC(CCOCCC)=O N1(C(CCCCC)=O)CC(CNC(C2(C)CC2)=O)OC(C)(C)C1 N1(C(Cc2scc(C)c2)=O)CCCC(F)(C(=O)NCC(N2CCOC2=O)C)C1 C1(F)(C(=O)NCCN(C(CC)C)C)CCN(C(c2cnc(O)n2CC)=O)C1 CCCC(C)(CC)C(=O)NC1CCCCCC1C(N1CCCC2(CC2)C1)=O Cc1ccc(COCC(=O)NC2CC2NC(=O)C(c2nc(C)cs2)C)cc1 C(=O)(CCCCCNC(N)=O)NC1CCN(C(C(CC)N(CC)CC)=O)CC1 c1(C(N2CC(N(C(c3cc(C)ncc3)=O)C)C(C)(C)C2)=O)cn(C)c(=O)cc1C CC1(C)CN(C(c2cocn2)=O)CC1NC(=O)C(F)=CC1CC1 C=CCC(C(=O)NC12CCC(NC(=O)CCSC3CCCC3)(CC1)C2)C(C)C CCCC(C)(C)C(=O)NC(C)C(CO)NC(C1CN(CP(C)(C)=O)C1)=O CC1(CCNC(c2cc[nH]c2C2CCCC2)=O)CCN(C(=O)COC(F)F)C1 C(=O)(CS(=O)(=O)N1CCCC1)NC(C1N(C(C(C)Cc2ccco2)=O)CCC1)C N1(C(Cc2c(C)n[nH]c2C)=O)CC(S(=O)(=O)N2CCN(C(=O)C=CCO)CC2)C1 C#CC1C(C(=O)NCC(C)(C)CN(C(=O)C=CC=CC)C)C1(C)C c1(C(N2CC(NC(CCCC=C)=O)C(C)C2)=O)ccc(Br)c(C)c1 C1(CNC(=O)CCF)CC2(CCN(C(c3ccc(C4CC4)cc3N)=O)C2)CO1 c1(C(=O)NC(CNC(c2ccc(C(N)=O)cc2)=O)CO)ccc2c[nH]nc2c1 N1(C(C2(OC)CCOC2)=O)CC(NC(C2CC(C(C)C)C2)=O)CC(F)C1 C(=O)(CCCCC(c1nn[nH]n1)N(C)CCn1cncn1)OC c1(C(=O)NCCCC(C)NC(=O)Cc2ccon2)cc2cccnc2nc1N Cc1c[nH]c(C#N)nc1=NC1CCCN(c2ccncc2F)C1 N1(C(Cc2ccc(C)s2)=O)CCOC2(CCC(NC(=O)CC(C)N(C)C)CC2)C1 C1(O)(CNC(C2(CC(C)C)CC2)=O)CC(NC(c2cnc(S)[nH]2)=O)C1 N1(C(C=CCOCCOC)=O)CCC(C(=O)NCC(C)(O)CCO)(OC)C1 S(=O)(=O)(c1ccc(Cl)cc1)NCC(=O)NC(c1nnnn1C(C)(C)C)C C1(CC(C)NC(=O)C(O)CC2CCOCC2)CCN(C(C2CS(=O)(=O)C2)=O)CC1 CC(C)(CCNC(C1CSCCS1)=O)NC(C1CCS1(=O)=O)=O c1(C(=O)NC2C=CC(CNC(c3n(C=C)ncc3)=O)C2)cc2c(s1)CCCCC2 C1(C(N2CCOC(CCO)C2)=O)C2C3CC4C1C2C34C(=O)NC(C)C(C)(C)C N1(C(C(C)=C(C)C)=O)CCN(C(C)=S)CC(O)C1.c1(C=O)conc1C(F)(F)F S(=O)(=O)(c1cc(Nc2c(C)c(CO)ccc2)c(Cl)s1)CN1CC2COCC2(CO)C1 C1(F)(C(=O)NCCCCCNC(c2cncc(C(F)(F)F)c2)=O)C2CCCCC12 c1(C(N2CCC(CNC(C3CC4CCC3C4)=O)C2)=O)cccc2ccncc12 C1(CC)C(NC(=O)Cc2cc(F)ccc2C)CCCN1C(c1coc(Cl)n1)=O c1(OC)cnccc1C(N1CCOC(C2CN(C(c3cc(C)n(C)c3)=O)C2)C1)=O c1(NC(C(CCC)C(C)C)=O)nc2ccccc2n1C(C1CCS(=O)(=O)C1)(C)C N1(C(c2ccc(CCC)cc2)=O)C2CCC1CC(NC(C1CSCC(=O)N1)=O)C2 C1(C(N2CCCC2C(=O)NCCC2CC3(COC3)C2)=O)CSCC(=O)N1 C1(CNC(C2CCc3n[nH]cc3C2)=O)(CBr)CC2(C1)CC(F)(F)C2 C#Cc1ccnc(C(=O)NC2(CC(=O)NC3(CCC=C)CCNC3=O)CCC2)c1 CC1CN(C(c2ccc(F)s2)=O)CC1CC(N1CCSC(C)C1)=O c12ccc(C(F)(F)F)cc1S(=O)(=O)NC1CN2CCO1.C(C(C)F)N(C)C C(=O)(C(C)=CCNC(=O)CCc1cocn1)N(CCC1CC1)CC CN1CCC(C(=O)NC2CCCCC2NC(=O)C=CSc2nc[nH]n2)C1=O CC(CS(C)(=O)=O)C(=O)N1CC2CC1CC2CNC(c1cnc(S)n1C)=O C(C(=O)NCCN(C(=O)C(F)(F)c1cncs1)C1CCCCC1)(C(C)C)SC c1(OC)nccc(C(N2CCC(NC(=O)C(C)(C)CC#N)CC2)=O)c1F C1(CNC(CCCC)=O)CN(C(c2cc(C3CC3)nn2C)=O)CCC12CCC2 C1(CC(=O)NC2CN(C(c3cnn[nH]3)=O)CC2C(F)F)CCC2(CC1)CC2 Cc1c(C(=O)NC2CCN(C(c3nccc(C(F)F)n3)=O)C2)sc(Cl)c1Cl CC1(C)OCc2c1n[nH]c2C(=O)NC1CCCN(c2nnc(-c3ccon3)s2)C1 C(C)(CCCCNC(c1c(C)coc1C)=O)NC(CCNC(=O)NC)=O C1(CNC(C(C)=C(C)C)=O)C2CCC2CN1C(C12CCCC1C2(F)F)=O c1(CC)[nH]nc(Cl)c1C(N1CCCC(CCNC(C2(SC)CC2)=O)C1)=O C(C(=O)NC(C)CC(C)NC(=O)CN1CCCCC1=O)(C(C)C)SC c1(OC)cc(C(=O)N(C(C)CNC(=O)CCc2cnoc2)C)cc(F)n1 c1(N2CCC(CN(C(C(OCC)OCC)=O)C)C2)nc(OC2CC2)cc(C)n1 C(=O)(C1=NN(CCO)C(=O)CC1)N(C1CCN(C(c2cc(SC)ncc2)=O)C1)C c1(C(CNC(C2(C=C)CCC2)=O)NC(=O)CC2CC3CC3C2)ccc(C(C)C)cc1 C(CC(CNC(C1C=CCCC1)=O)NC(c1ccsc1Cl)=O)OC Cc1c(CNC(C2CCc3nnnn3C2)=O)sc2cncn12 C(=O)(CCC(=O)N1CCC(O)CC1)N(C)CC1CCCN1C(c1cccnn1)=O C#CCC(C)C(=O)NC(C1CCCC1)CNC(c1csc(C2CCCC2)n1)=O C1(NC(=O)Nc2ccccc2)CCN(C(N(CC)Cc2cocn2)=O)C1 N1(C(C2(CC=C)CCOC2)=O)CCC(CNC(c2c(C)coc2C2CC2)=O)CC1 c1(C(N(CCCNC(C2(C)COC2)=O)CC)=O)ccc2ncc(Br)n2c1 c1(C(=O)NCC(=C)CCNC(=O)Cn2ccc(C(F)F)n2)cn(C)nc1CC C1(NC(C2C(C)CCS2)=O)CCN(C(=O)C=Cc2ccsc2Br)CC1 c1(CC(=O)NC(C)CCCNC(C2(C)CNC(=O)C2)=O)cnc2n1CCOC2 c12ccc(cc1)CC(=O)C2=O.C(=O)(CC(C)CF)NC1CC(C(C)=O)C1.CCCCN c1(C(N2CCCC(NC(COCCOCC#C)=O)C2)=O)cc(S(N)(=O)=O)cn1C C=CC(C)CC(=O)N1CC(CNC(c2cncc(-n3ccnc3)n2)=O)C1 Cc1ccc(CC(=O)NCC2CC2NC(c2nc(=N)cc[nH]2)=O)cc1Br N1(Cc2ccc(C(=O)OCC)n2C)CC(C)CS(=O)(=O)CC1 N1(C(c2n(CC)ccc2)=O)CC2CCCC2(NC(=O)CS(=O)(=O)NC(C)(C)C)C1 c1(C(N2CCC(C=C)(C(=O)OC)C2)=O)cnc2ccc(OC)nn12 C1(C(=O)NCCc2cccc(F)n2)CCC(F)(F)C1.C12(CCCC1)C(=O)N2 Cc1cc(O)c(C(=O)NCCC2CCN(C(c3nc(O)[nH]c(=O)n3)=O)CC2)nn1 c1(OC)cc(F)c(C(=O)NC(C)(C)CCNC(=O)CC2NC(=O)NC2=O)c(N)c1 c1(C(=O)NC2(CNC(C34C=CC(CC3)C4)=O)CC2)c(F)ccc2ccncc12 c1(C(CNC(=O)N(C)CC2CC2(C)C)(OC)COC)cc(C(F)(F)F)ccc1Cl C(CN=c1nc(-n2cccn2)cc(C)[nH]1)C1(OC)CN(C(=O)C(C)C)C1 c1(C(C(=O)NCC2CCN(C(C3(OC)CCC3)=O)C2)C)ccc(F)cc1F C1(NC(C(C)(C2CC2)OC)=O)CN(C(c2cnn(C3CCC3)c2C)=O)CC1C c1(C(=O)NCCC(C)(C)NC(C2C(C)(C)C2(F)F)=O)cncc2c(F)cccc12 CC1CCCCC1(CNC(c1ccc(CO)nc1)=O)NC(=O)CC(F)F O=C(C1CCCc2ccccc21)NCC1CCCN1c1ncnc2cccnc12 c1(CC)ccc(C(N2CC(NC(=O)C(C#N)C3CC3)C(C(F)F)C2)=O)cc1CC Cc1cc(C(C)C(N2CCN(C(C3(O)CCC(C)CC3)=O)CC2C)=O)cc(C)c1 C(=O)(CC(C(F)(F)F)c1ccon1)NCC1CC(OC)CN1C(=O)CO C1(CNC(c2n[nH]cc2C2CC2)=O)CC(O)CN1C(c1occc1Br)=O c1(C(C)C)ccc(N(CC(=O)NCC(F)CNC(=O)C=C2CCCC2)C)cc1 N1(C(c2c(CC)occ2C)=O)CC(NC(=O)C(F)C(C)C)CC12CCCCC2 CC1CCC(NC(=O)Cc2cnn(C)c2)CN1C(c1csnc1Cl)=O C(=O)(CC(F)(F)F)N(C(C)C(N1C2CCC1CC2)=O)CC c1(OC)cccc(C(N2CC(O)(CNC(C3CCCS(=O)(=O)C3)=O)C2)=O)c1OC c1(CNC(c2nnc(-c3ccccc3)s2)=O)cc(Cl)c(Cl)s1 C1(C(=O)NCC(CCOC)NC(C23CC(F)(C2)C3)=O)CC2(CCC2)CO1 C1(C(=O)NCC(N2CCCC2)C)CCN(C(C2C3CCCCC23)=O)C12CCC2 C1(C)(NC(C(C(C)(C)C)NC(c2ccn(C)n2)=O)=O)CCCCC1(C)C c1(CC(=O)NCCNC(CCCCC#N)=O)ccc2c(c1)CCC2 C1(NC(C=C(C)C(C)(C)C)=O)CCN(C(c2cc(C)cc(F)c2)=O)C(C)C1 c1(CC(N2CCC(F)(CNC(C(CCC)CC)=O)C2)=O)coc2ccc(C)cc12 c1(C(=O)NCc2n(CC)cnc2)cc2ncc(-c3ccc(C)cc3F)cc2[nH]1 N1(C(CNC(=O)OC)=O)CC(NC(C2(CC3CC3)CCC2)=O)CC12CCOC2 CC(C)C(F)(F)CC(=O)N1CCC(N(C(=O)CCn2cc[nH]c(=O)c2=O)C)C1 c1(C(=O)NCC2CN(C(c3c(OC)scc3)=O)C(C)CC2)cc(F)c(C)cc1O c1(C(N(CCN(C(=O)C(F)C(C)(F)F)C)C)=O)cc(O)nc(Cl)c1 C1(CC)(NC(c2ccc(C)c(O)n2)=O)CCCN(C(=O)COC(F)(F)F)C1 c1(C(=O)NC(c2cccc(OC)c2)CNC(=O)C=C2CC2)cc(C)nnc1O c1(OC)ccc(NC(N2C(C)CN(c3ccccc3)C2C)=O)c(C(F)(F)F)c1OC Cc1cc(C)c(C(=O)NCC2(CC(=O)NC(c3ncnn3C)CC)CC2)cn1 c1(CC(=O)NCC2CCCCN2C(C23CCCC2C3Br)=O)cc(F)cc(F)c1 C1(CC(=O)NCC2(CNC(=O)CC3CCCC34CC4)CC2)CCCC2(CCC2)O1 CC1CC2(C(=O)NCC3CCCN3C(c3cocc3C(N)=O)=O)CC12 C1(CNC(c2c(CC)n(C)nc2)=O)CN(C(=O)C(CO)OC)CC1(C)C CC(O)(CNC(=O)CCC1CCCCO1)CNC(=O)Cn1cnc(=N)[nH]1 CC1CN(C(C2CC(S(N)(=O)=O)C2)=O)CC(CCNC(C2CCCCC2)=O)O1 CCC(CC)(CN=c1[nH]c2cccc(F)c2o1)NC(=O)CCc1nc(O)n[nH]1 c1(C(=O)NCCN(C(c2c(C#C)c[nH]n2)=O)C)ccc(C)c2c1NCCC2 N1(C(c2cc(OC)n[nH]2)=O)CC(F)CC1CNC(=O)CC1CCCC(C)C1 C1(CNC(c2c(C)nncc2)=O)CC2(CC2)CN1C(=O)COC1CCCCC1C CC1CC2(CCN(C(c3cncc(CNC(=O)CC4CC5(CC5)C4)c3)=O)C2)CO1 Cc1cc(C(N2CCN(C(c3ncsc3C)=O)CC2CCO)=O)c2occc2c1 C1(CCSCCN(C(c2cnc(C)[nH]2)=O)C)CCCCN1C(=O)CN(C)C CN1CCC(C(=O)NCC2(O)CCOC2)(NC(c2cc(C(F)F)[nH]n2)=O)C1 C1(C(=O)OCC)(CNC(c2cnn(C(F)F)c2)=O)CCCO1.C12CC(C1)C2 c1(CNC(c2cc(CC(C)C)on2)=O)ccc(N2CCCOC2=O)cc1 C#CCCCCC(=O)N1CC=C(CNC(C2CCN(C(C)=O)C2)=O)CC1 c1(C(=O)NC(C)CC(C)NC(c2cnccc2Cl)=O)nc2cccnc2s1 C(=O)(C1c2ccccc2CN1C(c1ccc(C)nc1Cl)=O)N(CC=C)CC=C CCCC(C)(CCC)C(=O)NC1CCN(C(c2ccc(C3CC3)s2)=O)C1C N1(C(c2cccc(C)n2)=O)CC2CCC(N(C(=O)C(c3ccccc3)C)C)C2C1 c1(C(=O)NCC2C(C)CCN(C(c3cnccn3)=O)C2)ccc2scnc2c1 c1(C(=O)NC2C(NC(CCC)=O)CCCC2)cnn2ccc(Cl)c(F)c12 c1(C(N2CC(NC(c3c(OC)n[nH]c3)=O)C2)=O)c(C)nc(O)nc1C C(=O)(C(F)CC(C)(C)NC(c1ccc(F)s1)=O)Nc1ccc(COC)cc1 C1(CNC(c2c(Cl)cc(C)s2)=O)CC2CCC(C1)N2C(=O)C(c1cccnc1)O c1(SC(C#N)C2CC2)ccccc1.c1(C2C(=O)N2C)ccc(I)s1 C1(C(=O)NCC(C)OCC#C)CN(C(c2cc(CC)n(C)n2)=O)CC1(C)C C1(NC(CC2C(C)=NNC2=O)=O)CN(C(C2(CO)CC(F)(F)C2)=O)CC12CC2 c1(C(C)OC)nc(Cl)cc(=NCCCN(C(=O)CCCCSC)C)[nH]1 CCCC(C(=O)N1CCCC(CC(=O)NCC2CN(C(N)=O)C2)CC1)C(C)C C(=O)(C1=CCCC1)N1CC(C(N)=O)(CNC(=O)CCNC(C2CCCO2)=O)C1 c1(C(N(CCCNC(C2CC(OC(F)(F)F)C2)=O)C)=O)ccc(C(F)F)cc1F N1(C(c2c(C)cncc2)C(=O)NC2CCC2)CCC(C2=NOCC2)C1 CN1CCN(C(C2(CNC(c3ncccc3N)=O)CCC2)=O)C(CCO)C1 c1(C(=O)NC(c2cn(-c3ccc(Cl)c(F)c3)nn2)(C)C)occ2c1CCCC2 C1(NC(C2C(=C)C2)=O)CCC(NC(c2oc(CCC)nc2C)=O)CC1 CC1(CNC(c2ccc3c(c2)CCO3)=O)COCCN(C(C2CC3(CC3)C2)=O)C1 C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(c2cn(CCF)nn2)=O)C1(C)C c1(-c2ccc(C(=O)Nc3cscn3)o2)cccc(F)c1O.CC12CCCN1C2 c1(C(=O)NC(C(C)NC(c2[nH]nc(Cl)c2CC)=O)C(C)C)ccnc2cc[nH]c12 Cc1oc(-c2ccsc2)nc1C(=O)NC1CCC(NC(=O)CC2CC2(Cl)Cl)C1 C(=O)(C1CCc2cccnc21)N(CC(C)CNC(c1cccc(=O)n1C)=O)C c1(C(CC)(F)F)cccc(N(C2CC(C#N)C2)C(C2C(C(=O)OCC)C2)=O)c1 C1(NC(C(C)=CC2CC2)=O)(CO)CCCN(C(=O)C(C)n2ccnc2)C1 CC12CC3(C(=O)NCCOCCNC(=O)CCF)CC(C)(C1)CC(C)(C3)C2 N1(C(C2(C)CC(F)(F)C2)=O)CC2(CCCN(C(=O)CC3(N(C)C)CC3)C2)C1 c1(C(=O)NCCC(C)(C)NC(C2CC(C)OC2)=O)cc([N+](=O)[O-])ccn1 CC(F)(F)CCCC(=O)NC1(CF)CCN(C(C2CCCOC2)=O)C1 C=CCC(C(=O)N1CC(OCC2CC2)C(C(F)F)C1)OC1(C(=O)NSC)CCC1 CC1CN(C(c2c(N)cccc2F)=O)CCC1CNC(=O)CCCC(=O)C1CC1 CCC(CC(=O)NCC(C1CCCCC1)NC(=O)C(C(C)O)N(C)C)C1CC1 n1(CC)cc(C(=O)C(=O)NC2(CN(C(=O)C(C)NC=O)C)CC2)cn1 c1(C(N2CCN(C(CC(CC)C)=O)C(CF)C2)=O)cc(C)cc([N+](=O)[O-])c1N CC1CC(c2cccc(F)c2)N(N(C)Cc2ccc(Br)cc2)CCO1 C(C(C(C)C(C)C)NC(=O)CCCCCF)NC(c1ccc(N(CC)CC)nc1)=O Cc1ccc(C(CO)N(C(CC(F)(F)F)c2ccc(Cl)cc2)C)cc1 c1(C(c2n(C(CC)C)nnn2)NCc2ccnn2CC)ccncc1C C1(C(N(CC(C)(C)NC(c2ccc(C)s2)=O)C)=O)CC2(CC2)CO1 Cc1ccn2nc(C(=O)NC3CC4(CCN(C(C56CC(C5)C6)=O)CC4)C3)nc2n1 C1(O)(C(N(CCOCCOC)CCO)=O)CCc2cc(Br)ccc2C1 C(CCCCCNC(=O)C(C)(C)CO)NC(C1C(C)C1)=O N1(C(CC(C)OC)=O)CC(NC(c2ccc(Cl)c(OC)c2)=O)C(N=[N+]=[N-])C1 CC(C)(C#N)CCC(=O)N1CC(F)(F)CC1(C)CNC(=O)C=C1CCOCC1 c1(CNOCC)ccc(CNC(=O)C(C)OC(C2(NS(C)(=O)=O)CC2)=O)cc1 c1(N2CCC(O)C(C3CC3)C2)ncnc2cc(C(F)(F)F)ccc12 c1(OC)ccc2c(c1)CCC(N1CCOCC1CC(N)=O)C2 c1(C(=O)NC2CN(C(CC3CCC(C)CC3)=O)CC2O)cnc2[nH]ccc2n1 C1(NC(c2cc(CCC)nn2-c2ccccc2)=O)CN(C(C)=O)C2(CCC2)C1 C=Cn1nncc1C(=O)NCC(CC(=O)NCCc1cccnc1F)C1CCC1 C=CCC(CC=C)C(=O)NC1CCC(C)(CNC(=O)C(F)(F)CC)C1 c1(NC(CCNC)(C)C)nc2c(c(=NCc3ncc(Cl)cc3F)[nH]1)SCC2 c1(CCNC(C(C2CCCO2)NC(c2ccco2)=O)=O)ccccc1F c1(C(=O)NCCC(CC)(C)N)cccc2ccoc12.C(=O)(C(C)n1ccnn1)N c1(C(=O)NC(C2(O)CN(C(C3(Br)CC3)=O)C2)C)c(CN(C)C)cnn1C C(=O)(C1CCCc2nccn21)N1CCN(C(c2ccn(C)c(=O)c2)=O)CC1CF C(=O)(C(CO)NC(=O)Cn1ccsc1=N)NCC(C)CN(C)C.C(C)=O C1(CNC(C2N(C(CC3C(C)(C)OCC3)=O)CSC2)=O)CCC2(CCC2)O1 N1(C(C2(C)CCCO2)=O)CCCC12CCC(NC(=O)C=CC(N)=O)CC2 c1(CC)cccc(C(=O)NC(c2ccccc2)CNC(=O)CC2CC2(C)C)n1 c1(C(N2CCC(NC(=O)CCOC3CCC3)C2)=O)cccc(OCF)c1.C1(OCO)CC1 N1(C(C2(CC=C)CCN(C(C3(OC)CC3)=O)C2)=O)CC2CCCC(O)C2C1 C1(C(N(CCCCCCNC(C2(CO)CCCCC2)=O)C)=O)CCCCN1N=O C1(C(N2C(CNC(C3(C=C)CCCCC3)=O)CC(O)C2)=O)CCc2n[nH]cc2C1 c1(OC)cccnc1S(=O)(=O)NCC(C(=O)O)C1CCCCC1 N1(C(C2CCC(NC(C(C(=O)OCC)OC)=O)C2)=O)CCn2cnnc2C1C C=C(C)C(C)(C)C(=O)N1CCC(CCNC(c2c[nH]ccc2=N)=O)C1 Cn1ncc([N+](=O)[O-])c1N1CCN(C(=O)NCCc2cnn(C3CCC3)c2)CC1 C1(NC(C2(CC#C)CCCC2)=O)CCCCC1CNC(=O)CCOCC(F)F c1(C(=O)NCC(=O)NC2(CC=C)CN(C(C3CCCCC3)=O)C2)csc(C)c1N CC(C)C(C#N)C(=O)NCC(c1cc(F)cc(Cl)c1)NC(=O)OC(C)(C)C CC(C)C(O)CC(=O)NC1CN(C(=O)CC(C)C2CCCCC2)CCC1C(C)C C1(C(N(CC(CCC=C)O)C)=O)C(C2CC2)CCN1C(=O)C(C1CC1)SC C1(C(=O)NC(CSCC)(C)C(=O)Nc2ccc(Cl)c(O)c2)CC2(C1)CC(O)C2 CCCC(CCC)CCCC(=O)NCCCC(C)NC(C)=O CC1CCN1C(=O)COCCNC(=O)CNS(N)(=O)=O C(=O)(C1=C(C)OCC1)N1C2CC(NC(C3C(=C)C3)=O)(C2)C1 CCCCCC(C)CC(=O)NC1CC(NC(c2cc(Cl)nnc2O)=O)C1 C1(CNC(c2cnc(O)s2)=O)(NC(C2CC(CCO)C2)=O)CCOCC1 C1(F)(C(N2CCC(NC(c3c(C)oc(C(F)(F)F)n3)=O)C2)=O)CCC(F)(F)CC1 CCCCC(CC)C(=O)N1CCC(C)(C(N2CCOC(C)(C)C2C)=O)CC1 c1(C(=O)NC2(CF)CCN(C(c3c(C)ncn3C)=O)C2)cc2cccn2c(O)n1 CC1CCCc2ncc(C(N3CCN(C(=O)C(F)=CC4CC4)C(C)C3)=O)n21 CCCC(C)(C)C(=O)NCC(F)CNC(=O)Cn1nnc(C(C)(C)C)n1 c1(NC)cnncc1C(N1CCOC(C(C)NC(=O)CN2CCOCC2)C1)=O c1(C(=O)NC2CCN(C(CSCCC)=O)C(C)C2)cc(=O)n2ccsc2n1 O=C1CCCC(CC(=O)NC2CCOC(C(=O)Nc3c[nH]ccc3=O)C2)C1 C1(C(=O)NCC(C)Cn2cccn2)CC2(CC2)CN1C(=O)CN1CC2CC2C1 CCC(CC)CC(=O)N1CC2(CC(NC(C3SCCCS3)=O)C2)C1 n1(CCOC(c2cc(C)c(-c3cn(CN)nn3)cc2)=O)c(C)nc2ccccc12 c1(C(N2C3CC(CC(NC(CC(C)(C)SC)=O)C3)C2)=O)cccc2c1OCCO2 c1(C(=O)NCC(=O)N(CCCF)C)ccc(Br)c(Br)n1 c1(NC(=O)C2CC2)ccc(C(N(C2(CO)CC2)C)=O)cn1.C1(C(=O)N)CC(C(N)=O)C1 C#Cc1cccc(C(=O)N(C23CN(C2)C3=O)C)c1.C(C=C)C.C1(S)CC1 C1(CCOC)CN(C(=O)C(C)(C)O)CCN1C(c1cnc(C(C)C)o1)=O CC1CCSCCN1C(=O)CCCCN(C)C(C1CCC(=O)N(C)C1)=O N1(C(c2n(C)cnc2)C(=O)NCC2CCCO2)C2CCCC1CC(=O)NC2 c1(C(=O)NC2CCC(NC(C(C)=O)=O)C2)cccc(-c2ccccc2F)c1 C1(C)(CNC(c2cn(CC)nn2)=O)CCN(C(=O)C2=CC(C(C)(C)C)C2)C1 c1(C(=O)NCC2(F)CC(NC(CC3CN(C)C3)=O)C2)cc2c(F)ccc(F)c2[nH]1 C1(C)(CC(N2CC(CC(C)NC(c3cc(CO)[nH]n3)=O)C2)=O)CC1(F)Cl S(=O)(=O)(c1cnc(Cl)nc1)N1CC2(C(C(=O)NC(c3ccc(F)cc3)CO)C2)C1 CN1C(=O)c2ccccc2C1CC(=O)NC1CCC(NC(=O)Cc2ccsn2)C1 c1(C(=O)NC(CC=C)CNC(C2C3COCC23)=O)ccc2c(c1)CNC(=O)N2 c1(OCCOCCOC)ccc(N2C(=O)NC(c3cscn3)C2=O)c(C)c1 N1(C(C2C(C(N)=O)C2)=O)CCN(C(C2CCC2)=O)C2COCC12 C(=O)(C1=NOC(C)C1)NCC1CCC(NC(c2c(C)cccn2)=O)CC1 N1(C(c2cc(COC)on2)=O)CCC(N(C(c2cnc(C(F)F)s2)=O)CC)CC1 N1(C(C=CCN(CC)CC)=O)CC(NC(C2(c3cccnc3)CCC2)=O)C(C)C1 c1(C(N(C(C)C(=O)NC2CCC2)CCC)=O)cc(C)c(O)nn1 c1(COCC(=O)NCc2cc(OC)c(OC)c(C(N)=O)c2)nc(C)[nH]c1[N+](=O)[O-] C12(CNC(c3ccncc3Cl)=O)CCCC1CN(C(C1(C3CCCC3)CC1)=O)C2 N1(C(CC=C=C)=O)CCC(C)(CC(=O)NC(C)Cc2nncn2C)C1 C1(CC2(CNC(c3ccc[nH]3)=O)CCCO2)COCCN(C(C2CCCS2)=O)C1 Cc1ccc(C2CCNC2)nc1.C12CCC1CNC(=O)N2.C(C)(C)(C)OC(=O)NCC N1(C(c2c(OC)n[nH]c2)=O)CC(CNC(=O)Cc2cncn2C)C(F)(F)C1 N1(C(CCC)=O)CCCOC(CNC(=O)CSc2nccn2C)C1 N1(C(C2CCC(C)O2)=O)CCC(C)(CNC(=O)CCSc2ccc(F)cc2)CC1 C1(C(N(C2CC2)CC2N(C(C3CCC(CC)O3)=O)CCC2)=O)CCC(C)C(C)C1 C=C(C)CN=C(NCc1cnn(CC)c1)N1CCC(CC2CC2)C1 c1(CNC(CCOC(C)=O)=O)cc(C(=O)NCCCc2nncn2C)no1 C(=O)(C1Cc2ccccc21)N1CCC(=CCNC(CCC(C)O)=O)CC1 C1(C(=O)NCC(C2CC2)NC(COC(C)C)=O)CCc2ccccc2C1 c1(C(=O)NC(C(C)(C)C)CC(=O)NC23CC(CO)(C2)C3)ccc2oc(S)nc2c1 C(CCN(C)C)(C(=O)N1CC(O)C1)NC(C(C)SCCCC)=O C(=O)(C1COc2ccccc21)NCC1CCN(C(c2c(OC)ccc(Cl)c2)=O)C1 C(C)(C(O)C(=O)N1CC(CN(C)C(c2ccnc(-n3ccnc3)c2)=O)C1)SC N1(C2CCN(C(C3C(C=C)C3)=O)CC2)CCN(C(c2cn(CC)cn2)=O)CC1=O c1(C(=O)NC(C)CN2CCN(C(=O)CN(C)C)CC2)cn2ccsc2n1 c1(NCC2N(C(C3CCCCO3)=O)CCC2)nccc(-c2ccccc2F)n1 N1(C(C2(C(=O)OCC)CC=CC2)=O)CCCC(CNC(c2cc(=O)cc[nH]2)=O)C1 Cc1ccccc1C=CC(=O)NCC1CC1CNC(C1(C(C)(C)C)CCC1)=O N1(C(CNC=O)=O)CC(C(=O)NOCC(F)(F)F)C(F)(F)C1 c1(CN)c(C)cc(C)c(C)c1Br.C1(C(CN(CC)CC)C)CCOC1 C1(C(=O)Nc2ccc(C)cc2)CCCOC1(C)C C1(NC(CCCCC(C)C)=O)CCC2(CCCN(C(c3ccsc3)=O)C2)C1 C1(NC(CCC2N(C(C3CCCN(C)C3)=O)CCC2)=O)CC2(CCCCC2)C1 CC1OCCCC1C(=O)NC1CCCC1CNC(c1ncnn1C)=O C1(C(C)C)C(C(=O)NCc2nnc(C)o2)CCN1C(C1(N(C)C)CC1)=O C1(C)(CNC(C(c2ccccc2)OCC)=O)CCCN1C(c1cc(Cl)n(C)n1)=O CCC(C)(CNC(=O)CCC1CCOCC1)NC(=O)COC1CCC1 N1(C(=O)CC2CCC(F)(F)C2)CCOC2(C1)CN(C(c1cc(C(F)F)[nH]n1)=O)C2 c1(C(N(CCCCNC(c2cc(C#N)ccn2)=O)C)=O)cc2cccnc2cn1 N1(C(CN(C)CC)=O)CC(NC(=O)Cc2cnccn2)CC(F)C1 C1(C(C(=O)NC2CC(NC(=O)CCNC(C3CCCC3)=O)C2)O)CCOCC1 C1(C(=O)NC2CCC(C(N(C3CC(OC)C3)C)=O)C2)CC2(C1)CC2(F)F c1(CCC(N2CC(OC)C(NC(=O)C3=NNC(=O)C3)C2)=O)cc(C)nc(C)c1 C(c1cccc(CO)c1)=CC(=O)NCCCC1N(C(C2C(C=C)CC2)=O)CCC1 N1(C(CCC2CC(OC)C2)=O)CCN(C(=O)C(C)n2cccn2)CC1C1CC1 c1(C(=O)NCC(CNC(C2C(OC)CCC2)=O)(C)C)ccc2nnn(O)c2c1 C#CC1CC2(CC(C(=O)NCC3CCCN3C(=O)C(O)Cc3ccccc3)C2)C1 N1(C(=O)C=CI)CCC(C(C)(C)C)(CNC(c2cc(-c3ccccc3)ncn2)=O)C1 N1(C(CC2(C)CCN2C(c2cnnc(O)c2)=O)=O)CCC(O)(CC(N)=O)C1 Nc1ccc2c(c1)CCN(C(=O)CCc1cccc3ccncc13)C2 c1(CC(=O)NC2(C)CN(C(=O)COC3(C)CCC3)C2)c[nH]ccc1=O Cn1cc2c(CN=C(NCC3CCCO3)NCC3(C)CCCO3)cccc2n1 c1(C(=O)NC2CC(C(=O)NCCCOC)C2)c(F)ccc(F)c1OC C(C(C)(C)C(=O)NC1(C2CCCN2C(c2cncc(Br)c2)=O)CC1)OCC C(=O)CCCCCN(C(=O)CNC(=O)CN(C)C)C.C(C(CO)NC(C)=O)OC c1(C(=O)NCC2(C(=O)NCC3(O)CCCCC3)CCCO2)ncccc1O c1(C(=O)NC2C3CN(C(COCCCOCC)=O)CC32)cc(Cl)cc(Cl)c1 N1(C(C2CC(=O)CC2)=O)CCOC2(CCC(NC(c3cncs3)=O)CC2)C1 CCCCC(C)CCC(=O)N1CCC=CC1C(=O)NCC1CCC(=O)NC1 C1(N(c2cc(C)nn2-c2ccncc2)C(C2(Br)CC2)=O)CCNCC12CC2 C(C)(C(=O)N(C)CC1(CNC(=O)CSC)CCC1)SCC C(=O)(C(O)CC[S+](C)C)NC(C(C)C)(C)CNC(=O)CCN(S(C)(=O)=O)C c1(N(C)CC2(c3cccc(Cl)c3)CC2)cc(NCCc2cccc(F)c2)ncn1 Cn1nc(C(N)=O)cc1C(N1CC2C(CNC(=O)CC3C=CCC3)C2C1)=O CC(C)(C(=O)NCC=CCNC(c1ccc(=O)oc1)=O)C1=CCSCC1 N1(C(c2cn(CC3(C)COC3)nn2)=O)CC2(NC(C3(C(F)F)CCCO3)=O)CC1C2 c1(OC)cccc(Cl)c1CC(=O)N(CC(=O)OC(C)(C)C)CC1CCCO1 CC1CCN(C(=O)CCC2CCCCC2)CC1CNC(C1(F)CCOCC1)=O C1(CO)CC12CCN(C(=O)C(Cl)=CCl)CC2.C12CCCCN(C1)C(=O)CC2 CC(C)C(O)C(C)(C)C(=O)NCC1CCCC(CNC(=O)CC(F)(F)Cl)C1 C1(NC(C2=C(C)OCC2)=O)CCC2CC1CN2C(c1cc(Cl)ccc1N(C)C)=O C1(CNC(c2cncc(C)n2)=O)CCN(C(=O)CC2(N3CCCC3)CC2)CC1O c1(C(=O)NC(C)CNC(=O)Cc2cnnn2C)cccc(P(C)(C)=O)c1 C=C1CC(C(=O)N(c2ccsc2)C)(CNC(=O)C(O)CN2CCCC2)C1 C(=O)(C(C)(C)NC(=O)C1CC1)N(C)CCOCCCNC(=O)Cn1nccn1 N1(C(c2cc(C)ncc2C)=O)CCCC12CCC(NC(=O)Cc1cnns1)CC2 c1(N(CCC2CC(C)OC(C)C2)CC)c(C)cccc1[N+](=O)[O-] c1(C(N(C2C3CN(C(C4CCOC4)=O)CC23)C)=O)cncc(F)c1 Cc1nc2c([nH]1)CC(C(=O)NC(CO)C(C)NC(c1ccco1)=O)CC2 CCC(O)C(C)C(=O)N(CCCCCNC(c1ccc(OC)nc1OC)=O)C c1(CCC)ccc(C(C)NCc2nc(C(=O)NN(C)C)n[nH]2)s1 C1(C(=O)NCC(N2CCOCC2)C)(CC)CCCN1C(=O)CCN1CCOCC1 C1(c2cccc(CNC(C(CCSC)N)=O)c2)CCC2COCCC2O1 N1(C(c2c(CC)cc[nH]2)=O)CC(CNC(=O)C(C)CNC(=O)OC)C2(CC2)C1 N1(c2ncc(C)nc2)CCC2(CCCC(=O)N2)CC1 N1(C(c2c(C)sc(Br)n2)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1C CN1CCN(C(C2CN3CCC2CC3)=O)C(CNC(c2cnc(N)cn2)=O)C1 c1(-c2nc(CN(CCC)CCNC(C)=O)sc2)ccc2nc[nH]c2c1 C12(CC(=O)N(CCC)CCNC(=O)C(c3ccnn3C)O)CCC(CC1)C2 C1(C(=O)NC(C(=O)NCC=CCOC)C2CCC2)CC(O)CN1C N1(C(C2C3CCN(C(C(C)(C)O)=O)CC32)=O)CC2(C)COCC2(C)C1 CC(CS(C)(=O)=O)C(=O)N1CCOCC(NC(=O)Cc2cnn(C(C)(C)C)c2)C1 N1(C(CCCC(C)=O)=O)CC2(CNC(c3[nH]cnc3C)=O)CCC1CC2 C1(C(N(CCC)CCNC(c2cscc2CC)=O)=O)CCOC(C)(C)C1 C(=O)(C(C)C(C)S(C)(=O)=O)N(CC(C)NC(=O)CCN1CCCCC1)C c1(CCCC(=O)OCC)cc(=NC(C)c2ccnn2CC)[nH]c(C)n1 C(=O)(C1Cc2ccccc21)NCC1OCCCN(C(C2C(C)C2)=O)C1 CC1OCCC1(C)C(=O)NCC1CCC(C(=O)NCC2(O)CCOC2)CC1 c1(C(N2C(CNC(C3CC(C(C)C)C3)=O)CC(OC)C2)=O)ccc(C)c(F)c1F C(C)(N=c1[nH]c2c(c(=NCC(C)C(F)F)[nH]1)SCC2)c1ncc(C)cn1 Cc1cc(Cl)cc2[nH]c(C(N3CCC(N(C(=O)CC4CCOC4)C)C3)=O)cc12 C1(O)(CNC(C(C)OCCOCC)=O)CCCN(C(c2ccnc(OC)c2)=O)C1 c1(C(N2CC(CNC(C(CC)N3CCCC3=O)=O)C2)=O)cccc2c[nH]nc12 CC(C)(CC(=O)NCCCC1CCCCN1C(=O)CS(=O)(=O)C1CC1)C(F)(F)F N1(C(CC(C)(C)F)=O)CC(F)(F)CC1(C)CNC(c1cccnc1S)=O c1(C(N2CCC(F)(C(N(CCC#N)CC(=O)O)=O)C2)=O)cc(F)ccc1Br C1(C#N)(OC)CC(C(=O)NC(CC2CCCC2)C(=O)NC2(CO)CC(C)C2)C1 c1(C(=O)NC(C(C)NC(c2cc(C)c(C(N)=O)cn2)=O)C)cc2ccncc2s1 c1(C(=O)NCC2(CN(C(C(CCC)O)=O)C)CC2)ccc2cccnc2c1 c1(C(=O)NC2CN(C(CC=C=C)=O)C(C)CC2)ccc2ccccc2c1 C(=O)(CCCCCCCS(C)(=O)=O)N(CCOCCNC(CCC=C=C)=O)C C1(C(C(C)C)NC(=O)C(C)(C)C)CCCN(C(C2(Cl)CC2)=O)C1 Cc1cc(CCCNC(C23CC(C)(C2)C3)=O)on1 S(=O)(=O)(c1ccc(NC(C2(NC(=O)CNc3nccs3)COC2)=O)cc1)N(C)C CCC(CC1CCCC1)C(=O)N(C)CC1CN(C(C2(C)CCCO2)=O)CCO1 N1(C(c2cc(OC)no2)=O)CC=C(CCNC(c2csc3cncn23)=O)CC1 c1(C(CC(=O)NCC2(NC(C3CCOC3)=O)CCCCC2)CO)ccc(F)cc1 C1(CC(=O)OC)CCCN1C(C1CCC1(F)F)=O.C12(CC1)CC(=O)N2 C1(C(=O)OCCCCOC)CCC2(CCCC2)C1 Cc1ccc(C(C)NC(=O)CN(C(=O)CCc2cc(C)[nH]n2)C2CCC2)cn1 CS(=O)(=O)C(C(=O)NC1CN(C(=O)CCc2ncc(F)cn2)CC12CC2)C1CC1 CN1CC(C(=O)NNC(c2ccc(C#N)cc2F)=O)OCCC1=O CC1CC(C(=O)NC2CCCC2NC(=O)Cc2ccc(O)cc2C(F)(F)F)=NO1 c1(CN2C(C(=O)Nc3cc(C)sn3)CC(=C)C2)cc(F)c(Cl)c(F)c1 CC1C(C)N(C(=O)Cc2sc(S)nc2C)CCN1C(c1cc(C2CC2)cs1)=O N1(C(C(CN2CCOCC2)NC(C)=O)=O)CCCCC(C)(F)C1 N1(C(c2cn(C)c(=O)cc2)=O)CC2ON=C(CNC(=O)C3=NOCC3)C2C1 c1(C(=O)NC2(CNC(C3C(CC)C3(C)C)=O)CC2)ccc(C(F)C(F)(F)F)cc1 C(C(C)(C1CC1)NC(C1CC1C(F)(F)F)=O)NC(C=C(CC)C)=O C1(CC)(NC(=O)C(C)C2CCCC2)CCN(C(=O)C(F)C(F)(F)F)CC1 c1(OC)ccc(Br)c(C(N2CCCC(C)(CO)C2)C(=O)NC2CC2)c1 N1(OCC)CCN(CC(=O)NCCN(C(=O)Cc2ccccc2F)C)CC1 N1(CC)CCC(C(=O)NC(C2CCCN2C(C2CN(C(C)C)C2)=O)C)CC1 c1(C(=O)NCC(C)CNC(c2ccc[nH]2)=O)cc2cc(Br)cc(F)c2o1 N1(C(COCC)=O)CC(NC(c2cc(-c3ccc(C)cc3)n[nH]2)=O)C(CC)C1 c1(-c2ccc(C(N(C(CC)C(=O)OC)C)=O)cc2)ncc(C(F)(F)F)cc1OC C1(C(=O)NCC2(F)CN(C(C(F)=C(C)C)=O)C2)CCCC2(CCCCC2)C1 c1(CNc2cccc(C(=O)Nc3c(F)cccc3I)c2)ccc2c(c1)NCCO2 C1(NC(C2C(C)(C)C2CNC(C2(O)CCOC2(C)C)=O)=O)CCCCC1(C)C c1(CCC(=O)OC2CC3CC3C2)nc2cccc(Cl)c2[nH]1 Cc1nn(-c2ccc(F)cc2)c(C)c1CC(=O)NC1CC2C=CC1C2 c1(CNC(C2C3CN(Cc4c(C)ccnc4)CC23)=O)cc(NC(C)=O)ccn1 C=CCC(CNC(=O)C=CCCOC)C(=O)NC12CCC(C1)OC2C C(=O)(C(C)CC(C)(F)F)NCCN(C(c1nc(C)c(C)s1)=O)CC1CC1 Brc1scnc1-c1noc(C2CCNCC2)n1 C=CCC(CC(F)F)C(=O)N(C(C)CCNC(C1CCC2(CCC2)C1)=O)C N1(C(c2cncc(OCC)c2)=O)CCCC(O)(CNC(C2CC2C2CC2)=O)CC1 CC1CCCC(C(=O)NC(C)CNC(=O)CCn2cnnn2)O1 C1(O)(CNC(C=C(C)c2ccsc2)=O)CCN(C(=O)CC2(C)CC2F)CC1 C1(NC(CS(CC)(=O)=O)=O)CCN(C(=O)Cc2ncc(F)cc2Cl)CC12CCC2 C(=O)(CCCC(C)(C)C)N(CCOCCC(N1CC(CC)OCC1)=O)C N1(C(c2c(CC)cncc2)=O)CCCC12CCN(C(C1OCC1(C)C)=O)C2 C1(NC(CC2C(C)C2)=O)CCN(CCOC(C)=O)CC(C)(C)C1.C(C)(C)(C)O C12(C(N(CC(C)C(=O)NCCC(=O)NC3CC3)C)=O)CCCN(CC1)C2 N1(C(=O)NC(CC)CC2CCC(=O)N2)C2CCC1CC(F)C2 C#Cc1ccc(C(=O)NCCCC(CCC)NC(=O)C(C)CCOCC)nc1 N1(c2scc(C)n2)CCC(NC(C2CC2CNC(=O)OC(C)(C)C)=O)CC1 c1(C(=O)NC2C(CO)CCN(C(C(C(CC)C)C)=O)C2)c[nH]c2ncccc12 C1(C(N2C(C(C)(C)NC(=O)C(F)CC3CC3)CCC2)=O)CCC2CC2CC1 C1(NC(C(C(=C)C)(C)C)=O)CC2CC1CN(C(C1(C)CC1c1ccccc1)=O)C2 C(CN=c1nc(N2CCN(C)C(CO)C2)c2c([nH]1)CCCC2)OC N1(C(c2cc(CC)no2)=O)CCC(NC(=O)Cn2cc(C3CC3)cn2)C12CC2 c1(C(N2CC(CCNC(c3cnccn3)=O)OCC2)=O)n[nH]c2ccccc12 C=CCCCN=C(NC1CCCC1)NC1CCOC(CC(C)C)C1 Cc1c[nH]cc(C(=O)NC2CC(O)(CNC(c3cccn3C)=O)C2)c1=O Cc1cccc(C(N2CCN(C(=O)CC34CCCC3C4)CC2)=O)c1Cl C(Cn1ccnn1)(C(=O)N1CC(C(=O)OC)(CC)C1)NC(C=CC)=O C1(C(=O)NCC(CC)NC(c2ccc(N)cc2Cl)=O)CC(C)c2nc(C)cn2C1 CC1C(C)N(C(c2ccnn2CC#N)=O)CCN1C(=O)CCc1cccnc1Cl C1(C)(NC(CC(C)SC)=O)CCCN(C(c2ncoc2C(C)C)=O)C1 O(P(C)(=O)CCNC(=O)C(Cc1ccco1)NC(c1cc(OC)cnn1)=O)CC C12(C(=O)NCc3ccc(CC)s3)CC1CN(C(c1cccc(NC)c1)=O)C2 C(=O)(C1=CCCCC1C)N1CC(CC)N(C(=O)C(=O)N=S(C)(C)=O)CC1 c1(C(N(CCC(C(C)C)NC(C(CC=CC)C)=O)C)=O)cnc2c(c1)COC2 C(O)(CC(C(=O)NCCOC1CCOCC1)N(C)C)c1c(C)n[nH]c1 c1(NC(c2c(-c3cccc(OC)c3)cccn2)=O)cc(C#N)ccc1Br CCCCCCC(C)CC(=O)NC12CC(CNc3cnc(F)cn3)(C1)OC2(C)C CCC(C(=O)NCC=CCNC(=O)C(C)Cc1cnc[nH]1)c1ccccc1 Cc1nc(C=CC(=O)NCCCC(C)NC(C2CCN(C)C(C)C2)=O)[nH]c1C CCC(F)(F)CC(=O)NC1CC(C)(NC(c2ccc(Cn3ccnn3)cc2)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2CCOC2)=O)cc2cc(Cl)ccn2n1 C1(O)(CNC(C2(NC(=O)C(=O)NC(C3CC3)(C)C)CSC2)=O)CCCOC1 C(=O)(C1=CS(=O)(=O)CCC1)N(CC)Cc1ccc(-c2ccccn2)o1.c12cn-1nn2 N1(C(c2ccc3ncnn3c2)=O)CCC2(CCCN2C(C2CC2Br)=O)CC1 Cc1cc(C)c(C(N2CC(CNC(C3CCCN3N=O)=O)CC(C)C2)=O)c(O)n1 C1(NC(C(C)S(N)(=O)=O)=O)CCCC12CN(C(c1cnc(O)s1)=O)C2 N1(C(Cc2nc(C)[nH]n2)=O)CC2CCOCC2(NC(=O)CC2CC=CCN2C)C1 c1(C(C)C)ncc(C(=O)N(C2CCC(NC(c3cn(C(F)F)cn3)=O)C2)C)n1C C(=O)(C(C)S(=O)(=O)C(C)C)NC(CC)(C)CNC(C1(F)CCCCC1)=O C(=O)(C=C(Cl)Cl)NCCOCCN(C)C(C1(c2ncco2)CCC1)=O n1(-c2c(C)cccc2)[nH]nnc1=NC(=O)N(C(Cc1cncn1C)C(=O)O)C1CC1 Cc1ccc2[nH]c(CN3CCC4(CC4C(=O)NCCC(C)(C)O)C3)c(C)c2c1 c1(CC)cccc(NC(=O)CC2CN(C(=O)C(CO)NC(N)=O)C(C)(C)C2)c1F c1(NC2(CNC(COCCSC)=O)CCOC2)cc2ccccc2cc1C N1(C(C2C(CC(C)C)C2)=O)CCC(O)(C2(NC(=O)CCCCN(C)C)CC2)CC1 CN1CC(N=c2nc3sccc3c(N3CCc4ncccc4C3)[nH]2)CC1=O Cc1ccncc1CC(=O)NC1CN(C(c2cccnc2)=O)CC1C N1(C(CC2CC(C)C2)=O)CCC(C)C(CNC(=O)C=CC2CCCCCC2)C1 c1(C(=O)NC)cccc(C(=O)NCC2CC(NC(=O)Cc3csnn3)C2(C)C)c1 C(=O)(C(C)(CO)NC(=O)Cc1cccnc1O)N(C1CC2CC2C1)C C(=O)(CCCCC(C)(C)C)N1CCOCC(CNC(C2ON=C(C)C2)=O)C1 C#CCCCC(C)C(=O)NC1CC(CC(N2CCCCC2C(=O)NC)=O)C1(C)C N1(C(c2c(CC)[nH]cc2)=O)CC2(CC2)CC1CNC(c1nccc(OC)c1F)=O c1(OC)ccc(C=CC(N2CCC(C)C(NC(=O)C(O)C3CC3)C2C)=O)cc1Cl C(CC(C)(O)C(=O)NCc1cc(C(=O)NCCC(C)(O)C2CC2)no1)N(C)C c1(C(C(=O)NCC2(CCNC(=O)C(F)(F)CO)CC2)O)ccc(F)cc1F C1(N(C(CCCC)=O)C)CN(C(c2cc(C)n(-c3ccc(Cl)cc3)n2)=O)CC1O CCC(CC)CC(=O)N(C(C)CNC(=O)C(C)(C)Nc1ccccn1)CC N1(C(c2nc(C)sc2)=O)CCN(C2CCC(NC(=O)CC3(C)CCC3)CC2)CC1 N1(CCN(CCC)C(c2nccc(C)n2)C)CCC(c2nc(CC)no2)CC1 N1(C(C2C(C(=O)OCC)C2)=O)CCn2ncc(CN(C(=O)C(O)C3CC3)C)c2C1 CC1=NN(C)C(=O)C1CC(=O)NCC12CC(CN1C(c1ncccc1C)=O)C2 CCC(CC(=O)N1CC(C2CN(C(=O)CCc3cnc(C4CC4)o3)C2)C1)C(C)C C1(NC(CN(S(C)(=O)=O)C)=O)CCOCC1NC(=O)Cn1ncccc1=O c1(OC)ccnc(C(=O)N(C2CCN(C(=O)C(F)Cc3ccccc3)C2)C)c1 S(=O)(=O)(c1cccnc1NC(c1cn(CCCN(C)C)nn1)C)NCCCC=C N1(C(C(CC)F)=O)CC2CC(NC(=O)C(CO)NC(=O)OC(C)(C)C)CC1C2 N1(C(C2N(Cc3ncn(C)c3)CC2)=O)CCc2ncncc2C1 C(CCC)(CCCNC(=O)CN1CC(=O)NC1=O)NC(c1cnn(CC)n1)=O C1(C(=O)N(C(C)C(N)=O)C)(CC)CCCN(C(=O)CC#N)C1 C(=O)(C1=CC(C)(C)C1)N1CC(C(C)NC(=O)Cn2nccn2)C1 c1(C(=O)NCC(C(C)(C)C)NC(c2ccc(=N)[nH]c2)=O)cc([N+](=O)[O-])ccn1 C1(C(N2CCN(C(CCC#CC)=O)C(CC)C2)=O)CC2CCC(C1)N2C1CC1 C=CCCCCC(=O)N1CCCC(NC(C2CCCC(C(N)=O)C2)=O)C1 C1(NC(CC(C)OC)=O)CCCC2CN(C(c3ccc[nH]3)=O)CC12 N1(C(CSc2nc(C)[nH]n2)=O)CCC(NC(=O)CCCN2CCCCC2)C(O)C1 c1(C(N2CCC3C(NC(C=Cc4c(C)nccc4)=O)C32)=O)ccn2nnnc2c1 c1(C(N2CC(NC(CC(=O)NC)=O)C(OC)C2)=O)ccc2nnn(O)c2c1 C1(SC(C)C(=O)NC(C)(C)CN(C(=O)Cc2ccccc2)C)CCCCO1 c1(C(=O)Nc2sncc2C(F)(F)F)nccc2c1NCCC2 C1(CC(N2CCC(C(C)NC(=O)COc3ccon3)C2)=O)CCCCC1C c1(CC(=O)NC(CSCO)C)ccc(O)cc1.C(C(C)C1CC1)OC c1(NC(C2(OC)CC2)=O)ccc2c(c1)C(O)CC2 C(=O)(C1(O)CCCCCC1)NC1C(C)CN(C(=O)CCn2cnnn2)CC1 N1(c2nc(SC)nc(Cl)c2)CCC2(NC(C3CCC4CC4C3)=O)CCCC12 CS(=O)(=O)CC(=O)N1CC(CNC(c2cc(-c3ccccc3F)[nH]n2)=O)C(O)C1 N1(C(C2N(C(C(CC)COC)=O)CC=CC2)=O)CCc2nnnn2CC1 c1(C(=O)NCC(CC=C)NC(c2ccn3nccc3c2)=O)c(F)ccc(N)c1F C(=O)(C(CCC1CC1)NC(=O)CC(C1CC1)C1CC1)N(CC(COC)C)C C(CCN(C)C)(C(=O)N(CC(O)C(C)(C)C)C)NC(c1cc(OC)n[nH]1)=O CCC(O)C(C)C(=O)N1CCC(NC(c2cn(-c3ccccc3Cl)nn2)=O)CC1 N1(C(C(CC)NC(C2CCCN2C2CC2)=O)=O)CCCC(CC)C1 N1(C(C=Cc2c(C)ccs2)=O)CC(NC(=O)CCC2CC2)CC12CCC2 c1(CC(N2CCN(CC#N)CC2)=O)c(F)cccc1Br c1(C(=O)NC(C2CCN(C(=O)Cc3cc(C4CC4)on3)C2)C)nnc(S)n1C C1(CCNC(CC2(OC)CC2)=O)CSCCN1C(=O)CC(C)CF CC1CN(C(c2cnc(O)s2)=O)CCN1C(=O)Cc1ccc(C(F)(F)F)nc1 C(CC(C)(C)C)(C(=O)N1CC(O)CC1C(=O)N(C)CC1CCC(=O)N1)OC c1(C(=O)NCCO)cccc(O)c1.C(C)(C(=O)N1CCC1)OC Clc1cccc(CNC2CCCSC2)c1-n1nnnc1-c1ccccc1 Cn1ncc(C(=O)NC2CCOC(C(=O)NCCCC3CCC3)C2)c1Cl c1(C(=O)NC2C(NC(C(C=C)OC)=O)COC2)cncc(C)n1 c12ccc(cn1)OC(=O)C2.C1(NC=O)CCCC1CF.C1(COC)(CC2CC2)CC1 CCCC(C)(C)CNC(C1CCCN1C(=O)C(C1CCC(=O)N1)C)=O C=C(Cl)CC(C(=O)NC1CCOCC1C)NC(=O)C(C1CCC1)OCC n1(CC=C)nnnc1C(CCC1CCCO1)NCc1occc1C CC(C)C(C(C)NC(c1cnc[nH]1)=O)NC(c1cc(-c2ccc(Br)s2)on1)=O N1(CCC(=O)NCC(CN(C(=O)CC2CC2(C)C)C)O)CCC(O)CC1 N1(C(CC(=C)C)=O)CCCOC(CNC(c2nc(C(F)(F)F)cn2C)=O)C1 N1(C(c2ccc(C#N)s2)=O)CCCN(C(C2(C3CC3)CCCO2)=O)CC1CO c1(NC(C2(NC(C(C3CCCC3)OC)=O)CSC2)=O)csc(C(N)=O)c1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC2C(C(F)(F)F)CC2(NC(=O)C(C)=CCC)C1 N1(C(C(COCC)NC(=O)COC(=O)C2CC2)=O)CC2CCCC2(CO)C1 C(C(C)(CC)C(N)=O)NC(C(C)N(C(CCC(=C)Cl)=O)C1CC1)=O c1(C(=O)NC(CC)CNC(=O)CC(C)C2CCCCC2)cnc(C)c(Cl)c1 c1(C(=O)NCCC(CNC(c2cc(OCC)n[nH]2)=O)O)ccc2ncc(C)n2c1 C(CCCCC(=O)NCC1COCCO1)n1cc(-c2cccc(C)n2)nn1 N1(C(Cn2ncc(C)c2)=O)CC=C(C(C)(C)C(=O)N2CCC2CN=[N+]=[N-])C1 N1(C(C2(SC)CCC2)=O)CC(NC(c2ccc3[nH]ccc3n2)=O)C2(CCCC2)C1 CC(CNC(=O)CCC1CCCCN1C(=O)CNC(N)=O)CC(F)(F)F C(=O)(C1=NNC(C(F)(F)F)C1)NC1C=CC(CNC(c2c(C)ccnn2)=O)C1 C1(COC)CCN(C)C1.c1(C(N2CC3(C2)C(=O)N3)=O)nc(C)sc1C.COC Cc1nc(N(C)C)sc1NC(C1CC(C#N)C1)=O C(=O)(C1Cc2ccccc21)N1C(CN(C(C(CCC(C)C)F)=O)C)COCC1 c1(C(N(C(C)CNC(c2c[nH]c(=N)s2)=O)C)=O)cnn2ccccc12 N1(C(CCC)=O)CCC(CO)(CNC(c2cc(C)cc(Br)c2)=O)CC1 c1(OCC(=O)NCCC2(CNC(=O)CC3CCC3)CC2)ccc(Cl)cc1C#N C(=O)(C(O)C(F)(F)F)NCC1C(C)CCN1C(=O)Cc1nc(=N)[nH][nH]1 C#CCCCC(=O)NC(C(C)NC(c1ccc(CSCC)cc1)=O)C(C)C Cc1[nH]nc(C(N2CC(C3CCCCN3C(=O)CONC(=O)OC(C)C)C2)=O)c1F c1(C(C(=O)N(C2CC2)CC2N(C(CCC#C)=O)CCC2)C)ccc(CC)cc1 c1(C(N2CCCCC2)C)nnc(N2CCC(O)(C(F)F)C2)n1CC N1(C(c2ccc(I)c(F)c2)=O)CCC2(CC1)CC(C(N1CCC(CO)C1)=O)CO2 c1(C(=O)OC(N2CCC(c3cc(C)no3)C2)=O)cnc(O)c(C(F)(F)F)c1 C(c1ccnn1C)=CC(=O)N(CC(=O)NC1(C)CC(=C)C1)CCC CCC(C)(O)CNC(=O)C(COC(C)C)NC(=O)CCN1CCCC1=O c1(CC)cc(=NC(=O)CC(CC)N(C(=O)CC2CNC(=O)O2)C)[nH]n1C CC(C(=O)NC1CCCC(NC(C2CCC(F)C2)=O)C1)C(C)O Cc1cn(C)nc1C(=O)NNC=O.C1(F)CCCC1.C(C)(C)(CNC(=O)O)OC(C)(C)C CC1CC2(CCN(C(c3ccc(F)cc3Cl)=O)CC2)CN1C(=O)Cc1cc[nH]n1 Cc1cc(C(=O)NC2CC(CNC(=O)CC3(O)CCC3)CC2O)cc(C)c1F c1(C(=O)OCC)cc(S(=O)(=O)NC2(SNCC)CCCCC2)c(Cl)cc1Cl C1(N(C(=O)Cc2ccsc2)C)CCCC(NC(c2nnn(C)c2C(F)(F)F)=O)C1 N1(Cc2c(OC)ccc(OCC(=O)OC)c2)CCC2(CCCCN2C)C1 c1(CC(=O)NCC2(C)CCCC2NC(=O)Cc2cnoc2)ccc2ncsc2c1 c1(C(N2CC(NC(C(C)C(C)(C)C)=O)C(C(F)F)C2)=O)ccc2c(c1)NC(=O)C2 c1(C(=O)NCCc2ccc(C)cn2)coc2c1CN(C(=O)C1=CCCC1C)C2 CCC(CCC(=O)NCCOCCN(C(=O)CC(C)F)C)OC c1(C(=O)NC(CNC(=O)CCC2CCCCO2)CO)cc(O)ccc1Cl C=C1CCC(C(=O)NCC=CCNC(c2ccncc2NC)=O)CC1 C(=O)(CC(C)(C)F)NCc1cn(C2CCN(C(C3(CCCC)CC3)=O)C2)nn1 Cc1cc(F)ncc1CNC(=O)NC(C)COCc1ccccc1 CCCCC(C)N(C(=O)C(=O)N1CC(OCCOC)C1)C N1(C(c2c(C)cn(CC)n2)C(=O)NC2CCC2)CCc2c(cnn(C)c2=O)C1 n1(CC)cc(C(=O)NC(CNC(=O)COc2ccccn2)C(C)C)c(C(C)C)n1 c1(C(=O)NCC(c2cccnc2)NC(C2CC(=C3CC3)C2)=O)cnc(Cl)s1 c1(C(=O)NCC2(NC(C3OCC(C)C3)=O)CC2)ccc(S(N)(=O)=O)o1 C(c1cccc(F)c1F)=CC(=O)NCC12C(CN(C(C=CC)=O)C1)C2 N1(C(C2CCCN(C(COCCCN(C)C)=O)C2)=O)CC2(C1)OC(=O)NC2C CC1=NN(C)C(=O)C1CC(=O)NC1CN(C(=O)C(C)Oc2ccccc2)C1 N1(C(CC2ON=C(CC)C2)=O)CC2CCOC2(CNC(=O)C2=C(C)CCCC2)C1 CCCC(CNC(=O)C(C)OC)C(=O)N1CCC(n2ccnc2)C1 C(=O)(CS(=O)(=O)CCOC)N1C2CN(Cc3cccc(CC)c3)CC1C2 c1(CC(=O)NC2CCC(N(C(=O)CC3CC34CC4)CC)CC2)ccc(Cl)c(F)c1 C1(CC(=O)N(CCN(C(C(C(CC)O)C)=O)C)C)C2CC3CC(C2)CC1C3 C1(NS(CCOCC)(=O)=O)CN(C(c2noc(-c3ccccc3)n2)=O)CC1(C)C c1(C(=O)NC2CCC(N(C(c3occ(C)c3)=O)C)C2)ccn2ccnc2c1 C(C)(CCCCNC(c1ccc(Cl)cn1)=O)NC(C=CC(=O)OCCCC)=O C1(N(C(c2c(CCC)nco2)=O)C)CCCN(C(=O)C(c2ccccc2)F)CC1 CC1(C)C2CCC(C(=O)NCC3CCCC3NC(=O)Cc3cnc(C4CC4)[nH]3)C1C2 C1(C(CC)CC)CC(NC(=O)NC2(C(=O)OC)CS(=O)(=O)C2)CCO1 c1(OC)ccc(F)cc1NC(C1CN(C)CCN1Cc1ccccc1C#N)=O Cc1cc(C(=O)NC2(C(N3CCOC4(CC4)C3)=O)CC(O)C2)nc(O)c1 c1(C(=O)NCC2C(Cn3cc(CCn4cncn4)nn3)C2(F)F)ncccc1C c1(OC)ccc(CNCC2CN(C(c3ccc(F)c(F)c3)=O)CCO2)cc1C C(=O)(CC(C)(C)CC(F)(F)F)N1CC(NC(c2c(C(C)C)nns2)=O)C(C)(C)C1 C1(NC(CC2CCC(NC(C(CC3CC3)OC)=O)CC2)=O)CCC2(CCC2)C1 c1(C(=O)NCC2N(C(C(C)CC3CCC3)=O)CC(F)C2)ccc2ncsc2c1 C1(CN(C(C(C)O)=O)C)CCC(CNC(C2CC3(C2)CC3F)=O)CC1 N1(C(c2sccc2Br)C(=O)NCC(=C)C)CC(C)(C)c2cc(Cl)ccc21 CCCC(CC(=O)N1CCOCC1CCO)NC(=O)CC(C)CC C1(CNC(CCc2cc(OC)no2)=O)CN(C(=O)C2=CCC2)CCC1C(F)(F)F CCCCCCC(C)C(=O)NC(CNC(=O)Cc1c(F)cc(OC)cc1Cl)CC N1(C(C(C)OCc2ccccc2)=O)CCC(NC(C2CC2(F)F)=O)C2(CCC2)C1 c1(C(=O)NC2C(C)CCN(C(CCOC)=O)C2)ccc(O)c2ccccc12 c1(C(=O)NC2(C)CCN(C(C3CC(n4cnnc4)C3)=O)C2)cc2c[nH]cnc-2n1 C1(C(N(CC)CC2CCCCN2C(=O)C=C(C)C)=O)CCCCCN1C C(=O)(C1COc2ccccc21)NCCN(CC(C)O)C(C1C(C)(C)OC1(C)C)=O C1(C(=O)NC(C)CCNC(c2coc(C(N)=O)c2)=O)CCc2cnnn2C1 c1(C(=O)NCC2N(C(c3cc4nnn(C)c4s3)=O)CC2)ccc2c(c1)OCCO2 N1(CC)OCC(NC(C2CC(CCNC(=O)CC3CC(OC)C3)C2)=O)C1=O C1(NC(CC=CCC)=O)CCCC12CCN(C(=O)C(C)(O)CC(C)C)CC2 Cc1cccc(OCC(=O)NCCCCN(C(=O)CC2CCC(C)(C)O2)C)c1C N1(CCS(C)(=N)=O)CCC2(CC1)OCCc1cc(C(=O)NCCCO)sc12 N1(C(C(C)(C)CCl)=O)CCOC(C)(CNC(C23CC=CC(C2)OC3)=O)C1 C1(C)(CNC(C(C2CCCC2)OC)=O)CN(C(=O)Cc2ncoc2C)CCO1 c1(C(=O)OC)c[nH]c2ncnc(N3CC4CN(C(c5cccnc5)=O)CC4C3)c12 CC(C(=O)N1CC2C(NC(C3CC(=C4CCC4)C3)=O)C2C1)C1=CCCC1 c1(C(=O)NCC(C2CCCN2C(C2CNC(=O)O2)=O)(C)C)cnn(CCO)c1N c1(C(N(CCCOCCN(C(Cc2nc(CC)sc2)=O)C)C)=O)ncn(C)c1C N1(C(c2c(C(F)F)ccc(C)c2)=O)CC2(CCC(CNC(=O)C(C)O)O2)C1 N1(C(C(C)=CC2CC2)=O)CC2(NC(c3ccc(C)nc3O)=O)CCC1C2 Cn1cc(NC(c2cc(CNC(C3CCCN3C3CC3)=O)[nH]n2)=O)c(C#N)n1 C1(C(=O)NCC(C)CC(F)(F)F)CN(C(=O)C(c2cccnc2)N)CCC1O c1(C(=O)NC(CC=C)CC(=O)NCc2cnc(C)nc2C)cc2ccccc2[nH]1 c1(C(=O)NCC23CC(NC(C(CC=CC)C)=O)(C2)C(C)O3)cn2ccccc2n1 N1(C(c2cnc(CCC)s2)=O)CCC(CCNC(c2cnnn2C(C)C)=O)CC1 c1(N(C)C)ccc(C(=O)NC2CC(NC(C3(CCF)CC3)=O)C(O)C2)cn1 c1(C(N2CCC(NC(c3cccnc3OC(F)F)=O)C2)=O)ccc(Cl)c(Cl)c1O C(=O)(C(C)(C)NC(=O)NC1CC(C(=O)N(C2CC2)Cc2ccccc2)C1)OC CC(C)CC(C(=O)NCC1CC(NC(c2ccc(C(C)C)o2)=O)C1)C(C)C C1(C(=O)NCC2C=CCN2C(c2cnc[nH]2)=O)(OC)CCSC1 c1(N(C)C)ccccc1C(=O)NCC1CCCC1NC(=O)CC1(C2CC2)CC1 C1(C(=O)N(CC(C)C(=O)OC)C)(OC)CCN(C(c2coc(C(N)=O)c2)=O)C1 N1(C(c2cc(CC)n(C)n2)=O)CC(NC(c2ccccn2)=O)C(C)(C)C1 C(=O)(C(CCSC)N(C(=O)C(C1CCCC1)OC)C1CCOC1)OC CCCCCCC(C)CC(=O)N1CCC(CO)(NC(=O)Cn2cnnc2O)C1 c1(C(C)C(=O)NC2CCCN(C(C3(C)CC(C)(C)C3)=O)C2)cc2ccccc2s1 Cc1cc(C(=O)NC23CC(NC(=O)C4=NNC(=O)C4)(C2)C3)c(F)cc1Cl c1(NC(Cc2cc(C)on2)=O)ccc(C(C)N)cc1.c1(S)ccc(Br)cc1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(CC)N(C(C2CCC(C(N)=O)CC2)=O)CC1 C12(CNC(CC(C)(C)OC)=O)CCCC1N(C(=O)C=C(C)C1CC1)CCC2 Cc1ccc(CN(C(=O)COCCCN=[N+]=[N-])CC23CCC(CC2O)C3)c(O)c1 C1(NC(C2(CSC)CN(C(=O)CN3CCOCC3=O)C2)=O)(CO)CC2CCCC12 C1(C(=O)NCCN(C(C2(CC#C)CCOCC2)=O)CC)CCCC(C#N)C1 Cc1cccc(CNC(C2CC(C)CN(C(=O)CCNC(=O)CO)C2)=O)c1F N1(C(C2CCCC(C)O2)=O)CC(C2(NC(c3ccsn3)=O)CC2)C1 C1(c2nnnn2C(C)C)(Nc2cccc(NC(CCC)=O)c2)CCN2CCCCC12 c1(CNC(=O)NC2CC(=O)N(CC(CCO)C(F)(F)F)C2)cc(Cl)ncc1F c1(C(=O)NC(CC)(C)CNC(=O)C=Cc2ccnn2C)cncc2cnccc12 N1(C(c2c(F)ccc(C#N)c2)=O)CC=C(c2cccc(Cl)c2)CC1 Cc1ccc(CCCC(N2CC(NC(c3ccn(C)c3)=O)CC2C)=O)cc1 c1(C(N2C(CNC(c3c(C)noc3)=O)CC3CC32)=O)cc2c(Br)cccc2[nH]1 c1(N(CC(=O)N(Cc2c[nH]nc2C(F)F)CC2CC2)C)nc2ccccc2o1 S(=O)(=O)(c1cnccc1N(C)CC1CCS(=O)(=O)CC1)NCC(C)OC(F)F N#Cc1ccccc1-c1nc(C(=O)NCC(N2CC(F)(F)CC2C)=O)ccc1F C1(C(C(=O)NC2C(CNC(CNS(NC)(=O)=O)=O)CC2)O)CCS(=O)(=O)CC1 C1(NC(C2C(COC)C2)=O)CCCCN(C(c2ccc(F)cc2N)=O)C1 c1(C(=O)NCC(N2C(c3nnc(C)o3)CCCC2)=O)cn2nccc2nc1C c1(OC)ccc2c(c1)CC(C)N2C(=O)CCCc1cncc(Br)c1 c1(NC(C2CC2C=O)=O)oc(CO)cc1C.C1(C(=O)NCC)CC(C(=O)OC)C1 C1(C(=O)NC(c2nn[nH]n2)CC)CSCN1C(=O)C=CC(C)C C(=O)(C1CCCc2c(O)cccc21)N1CC(CN(C(C=C(C)Cl)=O)C)C2(C1)CC2 C#Cc1ccc(C(N2CCC(NC(=O)CCc3c[nH]c(=N)[nH]3)CC2C)=O)nc1 C(C)(C(=O)NCC1(CC(=O)N(CC(O)CC)C2CC2)CC1)OCCOCC N1(C(c2c(C#C)c[nH]n2)=O)CC(O)CC1(C)C(=O)NC1(CSC)CC1 Cc1cc(Cl)cc(C)c1C(=O)NC1CCCC1CNC(=O)CCCc1cc[nH]n1 c1(C(C(=O)NCCNC(c2ccn(CC(C)C)n2)=O)O)ccc(Cl)c(Cl)c1 N1(Cc2cn(CCCNC(c3c(C)c(C4CC4)on3)=O)nn2)CCCC(C)(O)C1 C12CN(CCC1(C)C)C2=O.c1(C(=O)OC)ccc(=O)n(CC2CCC2)n1 N1(C(c2c(O)cccc2Cl)C(=O)NCC(F)F)CCS(=O)(=O)C2(CCCC2)C1 N#Cc1ccc(O)c(C(N2CCC(NC(=O)Cc3cccc(Cl)c3)C(O)C2)=O)c1 N1(C(C2(CN(C)C)CC2)=O)CCN(C(c2c(F)cc(O)cc2F)=O)CC(CO)C1 C(C(C(=O)NCC(N1CCCC1)C)NC(=O)C(C)c1ccco1)OC(C)C N1(C(=O)NC(COc2c(CC)cccc2)(C)C)CCN(C(C)=O)C(C)C1 c1(NCC)ccc(Cl)cc1C(=O)NCC#CCNC(=O)CCc1cn[nH]c1 C1(CC(N2CCC(C(N(CC#C)CCOC)=O)C2)=O)CCC(=O)N1C N1(C(CNC(c2cccs2)=O)=O)CCOC(NCc2ccnc(C(F)(F)F)c2)C1 C1(NC(c2cnc(CC)s2)=O)CCCC(NC(c2cccn2CC)=O)C1 CC(CCCNC(=O)CC1CCCN1C)NC(=O)CN(C1CCC1)C C(=O)(C(C)(C)CCC#N)N(CCNC(C1CC(CC(=O)OC)C1)=O)C(C)C CP(C)(=O)C(O)C(=O)N1CC2CC1CC2NC(c1coc(C2CC2)n1)=O C1(C(N(C(C)C(=O)NCCc2noc(C)n2)CC)=O)CC2(C1)CC(C)C2 CCC(C)C(CC(=O)NCC(O)C(C)(C)O)NC(c1cc(C)sn1)=O CC(C)(C(=O)NCC(CO)NC(=O)CC1CC=CC1)c1cccnc1 c1(C(=O)NCC(CNC(c2c(C)csc2)=O)(C)O)cc(S(N)(=O)=O)cn1C c1(NC(C(=O)N(C(C)CS(C)(=O)=O)C)=O)ccc(Br)nc1Cl N1(C(C2(COC)C=CCN2C(=O)CC2CCCOC2)=O)CCC(C)CC1C C1(NC(C2(COC)CC=CCC2)=O)CCN(C(=O)C(C2(O)CCCC2)F)CC1C N1(C(C2C(c3c(C)cccc3)C2)=O)CCC2(C1)CN(C(c1cccs1)=O)CCO2 C(=O)(C1COc2cc(C)c(C)cc21)NC1(CNC(CC=CC=C)=O)CCC1 n1(CC(N2CC(C)(NC(C(n3cc(Cl)cn3)C)=O)C2)=O)ncc(Br)c1C C(=O)(CC(=O)NC(CO)C(=O)N1CCC1(C)CCO)N(C)C C(=O)(C1=CCOCC1)N1CCC(C(=O)NC(COC)CO)(OC)C1 C1(F)(C(N(CC(CC)O)C2CC2)=O)CCN(C(C2(C)CC3(CCC3)C2)=O)CC1 C1(C(C(=O)N(C(C)C)CCF)NC(C2CN(C3CCC3)C2)=O)CC=CCC1 C1(NC(C2CC(CCC)OCC2)=O)CCN(C(=O)C(C2CC(F)(F)C2)O)C12CC2 C(=O)(C(O)CCCc1ccccc1)NC(CNC(c1ncc(C)nc1)=O)CO c1(C(N2C(CC(=O)N(C)Cc3ccccc3)CCC2)=O)c(Cl)cccc1Cl C1(C(=O)NC(C#C)C)CCN(C2CCN(C(=O)C3CC3)CC2)CC1 c1(C(=O)NC(C2(CNC(CCOC)=O)CC2)C)c[nH]c2nc(Cl)ccc12 c1(C(n2c(-c3ccc(-c4c(F)cccc4Cl)s3)nnc2S)C)ccc(F)cc1F C#CCC(C(=O)NC(C)C(C)NC(=O)CN(C1CCCC1)C)C1CC1 c1(NC(C(C)NC(=O)NCCOCC(F)(F)F)=O)cnc(CC(=O)O)[nH]1 N1(C(c2c(C)cnnc2)=O)CCC(C)N(C(=O)COc2ccc(O)cc2)CC1 c1(OC)cc(C(O)C(=O)NC2CCCN(C(=O)C(F)=C3CCC3)C2)c(F)cc1O C(C(C)(C)CC(C)C)NC(C(CCC1CCC1)NC(CC1C(NC)C1)=O)=O O=C(CC(C(F)(F)F)n1cccn1)NC1COC2CN(C(=O)C(F)(F)CO)CC12 NS(=O)(=O)c1ccc(C(=O)NC2CCC(CNC(c3nncs3)=O)C2)nc1 C1(NC(c2cnn(-c3ccccc3)c2)=O)CCN(C(C2(CC(F)F)CC2)=O)C1 CCCCC(O)C(C)C(=O)NC1(CC(=O)Nc2cc(F)ccc2F)CC1 C12(C(=O)NC(CNC(CCSCC(N)=O)=O)C3CC3)CC(F)C1C2 N1(C(C(CCC)C)=O)CCOC2(CCN(C(C34CCCC3CCC4)=O)CC2)C1 c1(C(=O)OCC)cccc2nc(C(=O)N(C)C(C3CCCCC3)C)cn12 N1(C(C)Cn2cc(CSc3ccnc(Cl)c3)nn2)CCC(c2n[nH]c(=N)o2)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC(O)C(C)C)NCc1c(C)ocn1 C(=O)(C(C)C(O)C(C)C)NC1(CF)CCN(C(C(Cc2c(C)cccc2)C)=O)C1 C1(C(=O)OC)CCN(C(=O)C(=O)Nc2cc(C)n(C(C)C)n2)C(c2cccs2)C1 N1CCC(C)(CN(CCO)CC)CC1.C(C(F)C=O)N(CC)CC Cc1c(C(=O)NCc2ccc(C(F)(F)C(F)(F)F)s2)cnn1C(C)(C)C N1(C(c2c(C)nsc2)=O)CCC2(CCN(C(C34CCCC3C4)=O)CC2)C1 C1(NC(C=CCN(C)CC)=O)CN(C(c2cncc(C)c2)=O)CC1S(C)(=O)=O c1(NCC(=O)N(CC(C)CNC(=O)C=CCC2CCCO2)C)ccccn1 c1(OC)cc(C)cc(F)c1CNCC12CC1CN(C(=O)OC(C)(C)C)C2 c1(C(N2CCCC(N(C(=O)C=C3CCCCC3)C)C2)=O)cccc(P(C)(C)=O)n1 c1(C(=O)NC(C(C)C)C(C)NC(C2(O)CC(F)(F)C2)=O)cn(C)c(=O)n(C)c1=O N1(C(c2cccc(C(C)(F)F)n2)C(=O)NC(C(=O)OC)C)CCC(C)OC(C)C1 N1(C(c2ccc(CSCC(C)C)o2)=O)CC2C(CNC(C3CC3F)=O)C2C1 c1(C(=O)NCC(CNC(=O)C(O)C2CC2)OC)cc([N+](=O)[O-])c(Cl)cc1Cl c1(C(=O)NC(CCOC)CNC(=O)C(C)c2cccs2)ccc(S(N)(=O)=O)s1 C1(C(=O)NCC(CCNC(C2(NC(N)=O)CC2)=O)O)OCC2COCCC12 C(=O)(C(C(C)(C)C)C1CCC1)N1C(CN(C)C(c2cccnc2)=O)CCCC1 c1(C(N(CCN(C(CC2C(C)CCC2)=O)C)C)=O)ncccc1S(C)(=O)=O N1(C(COC(CC)(C)C)=O)CCN(C)C(C(=O)NCC2CCOC(C)(C)C2)C1 c1(SCC)cc(C)ccc1C(=O)NCC1CC(O)CN1C(=O)CC1CCC1 CCC(C)C(O)C(C)C(=O)NCC(C(=O)NC1CC(=O)N(O)C1)C(C)C C1(F)(CNC(c2c(C)scc2)=O)CCN(C(C2CCNC2=O)=O)CC1 C(CN=C(NCCSC)NCC(c1ccccc1)(C)O)c1ncc(C)cn1 c1(OC(c2c(CCC)n(CC)nn2)=O)cnc2n1CCCC2 c1(CCC(N2C(CNC(C(CC)=CCCC)=O)CC2)=O)ccccc1NC(C)=O CCCN=C(NCc1ccc(C)c([N+](=O)[O-])c1)N1CCC(C(C)O)C1 N1(C(C(C(C)O)NC(C(C(CC)C)N(C)C)=O)=O)CCC2(CC=CCO2)C1 C1(C(=O)NC23CC(C(=O)OC)(C2)C3)CC2CN(C(C3CN(C)CCO3)=O)CC2C1 C1(NC(c2c(CNC(C(C)n3cnnn3)=O)cnn2C)=O)CCN(C)CC1(C)C Cn1cnc2sc(CNC(N3CC(CNC(=O)OC(C)(C)C)C(O)C3)=O)cc12 c1(OC)cccc(CN(C2C(C)CNCC2C)C)c1C C(=O)(C1=C(CC)N(C)C(=O)NC1c1nc2ncccn2n1)OCC CCCCC(=O)C(=O)NCCC(C)CCNC(=O)CNC(c1ccccc1C)=O c1(CC(=O)NC(C)CNC(=O)C=CC(N2CCOCC2)=O)ccc(S(C)=O)cc1 c1(C(=O)N)ncc2ccccc2c1O.C1(C(=O)OCC)(C(=O)NC2CCCC2)CCC1 c1(CC(=O)N(C(C)CNC(=O)Cc2csc(C(F)(F)F)n2)C)cccc(F)c1Cl c1(C(=O)NCCC(C)N(C(C=CCOC)=O)C)cccc2c1OCC2 C1(C(=O)NCCCc2ncn(C)n2)CN(C)NC1=O O=C(CCC(=O)N1CCC(O)CC1)NCCC1(NC(C2CC(F)C2)=O)CC1 c1(C(=O)NC2C(C)(C)CN(CC(=O)NCc3ccccc3)C2)cc2ccccc2[nH]1 C(C1=NOC2COCC12)NC(N(C(CC1CC1)CC(C)C)CC)=O c1(NC(CC2CCN(C(c3scc(C)c3)=O)CC2)=O)cc(F)cc(C)c1Br c1(NC(C)=O)ccc(C(N2CCC(c3ccccn3)CC2)=O)cc1F c1(C(N)=O)n[nH]c(=NC2CCN(C(C3CCCS(=O)(=O)C3)=O)CC23CCC3)s1 C(=O)(C1=CC2CCCCCCCC12)NC(C(=O)N(c1cccc(OCC)c1)C)=O C(=O)(CC(CC(=O)O)C(F)F)NCCCC1C(C)C1 C1(C(=O)N(C(C)C(N2CCC(OC(C)C)CC2)=O)C)(CC)CC(C)(C)C1 C=CCC(CC=C)C(=O)NC1(C(=O)NCCCC(=O)NO)CC1C O=C(C1=C(Cl)CCOC1)NC1CCCCC1NC(c1ccc2nc[nH]c2n1)=O C1(NC(=O)C=C2CCOCC2)COC2CN(C(C3(CC4CC4)CCC3)=O)CC12 C=CCCC(C(=O)NC1CCOCC1)N(C1CCCCCC1)CCN(C)C C1(CNC(c2n(CC)c(O)nc2)=O)CCN(C(c2cc(=N)[nH]n2C)=O)CC1C c1(C(=O)NCC(=C2CN(C(=O)CC3(CO)CC3)C2)F)cc2cc(Cl)ccc2o1 c1(NC(=O)NC(C(=O)OC)CC2CC=CCC2)ccccc1CO.c1cccnc1 c1(OC)ccc(NC(=O)NCC2CCCC(C)O2)cc1F CCC1C(=O)NC(C)C(=O)NCC(=O)N1C.C(=O)(C(C)C)NCC1CC1 C(=O)(C1=NOC2(CCC2)C1)NCC1CCN(C(C(CC(C)C)OC)=O)C1 c1(CN2CC(CS(=O)(=O)N(C)C)NCC2)cc(Cl)cc(Br)c1 c1(N2CC(COC)SCC2)cc(C)[nH]c(=NCCCCCC(=O)N(C)C)n1 c1(CC(=O)NC2C3CN(C(C(CC=C)(C)C)=O)C(C3)C2)cnc2c(C)cccn12 S(=O)(=O)(c1cnc(NC(C)(CO)CCF)c(Cl)c1)NC(C)COCC1CC1 N1(C(C(COC)(C)C)=O)CC(C)CN(C(c2cnc3ccncc3c2)=O)C(C)C1 C1(NC(CCn2cc(-c3cn(C(C)C)nc3)nn2)=O)(CO)CCC(C)(C)C1 CCC(C(=O)N(CCCCO)CC)NC(N)=O N1(C(c2c(CC)nc(C)nc2)=O)CCCC2(C1)CN(C(=O)CSC(C)C)CCO2 CCC(C)C(O)CC(=O)N1CCOCC(NC(c2ccc(C)c(C)n2)=O)C1 c1(C(=O)NC2(COC)CCNC2=O)coc2c1CN(C(=O)C1CC1)C2 C#CC1(CNC(=O)CCN(C(c2cncc(C)c2)=O)C(C)C)CCCC1 C1(C)(C(N(CCC)CCNC(=O)Cc2n[nH]cc2Br)=O)CCSCC1 Cc1cc(C)n(C)c(=O)c1C(N1CC(NC(=O)CCF)CCC(O)C1)=O C12COCCC1C(=O)N(CC1CC1)C2=O.CC1(C)CCC1CCCN1CCCC1 n1(CC)c(C(=O)NC2CCC(F)(CNC(=O)COC3CCCCC3)C2)cnc1O Cc1nc(C(=O)NCC2CCN(C(C3CCCN3C3CC3)=O)C2)cc(O)n1 N1(C(c2n(CC)c(O)nc2)=O)CCN(C(C2(CCF)CCOCC2)=O)CC(O)C1 CC1CCCC1C(=O)N(CCCOCCNC(=O)C(C)n1ccnc1)C C1(C(=O)NC(C(C(C)C)O)C)CCCCN(C(=O)Cc2nc(=N)[nH][nH]2)C1 c1(C(N(C(=O)CN2CCC(n3cccn3)C2)C)=O)cccc(-c2cccs2)c1 c1(CN)cn2ccc(C(=O)Nc3cncc(CN4CCNCC4)c3)cc2n1 c1(N2C3C(NC(CC(CC)C4CC4)=O)(CCC3)CC2)ncnc2c1cnn2C C1(C(N(C)C)=O)CCCCN1C(C1CC(O)CN1C(=O)N(C)C)=O.C1(O)(C)CC1 CC(C(C)NC(=O)Cc1csc(NC(=O)C2CC2)n1)S(C)(=O)=O N1(C(=O)Cc2cccc(O)c2)CCC2CN(C(=O)C3=CC(O)CCC3)CC2C1 CCC(O)C(=O)N(C)CCN(C(=O)CC1CCCOC1)C N1(C(CN(S(CC)(=O)=O)C)=O)CCOCC1CNC(=O)C=C1CCN(C)C1 c1(CCC(N2C(CNC(CC3CCCN(C)C3)=O)CC2)=O)cc(Cl)ccc1Cl N1(C(COCC)=O)CCCC(C)(C)C1CNC(=O)CC1(C)CCOC1 C1(C(N2CC(C(C)NC(c3cnn(C4CCCC4)c3)=O)C2)=O)CC2CC1C1CC21 c1(OC)ccc(CCC(=O)N(C)CC2CCCN2c2nccnc2F)cc1 C1(C(C)NC(=O)C(c2ccon2)N(S(C)(=O)=O)C)CCCN1Cc1ccncc1 C(=O)(C(C)C(O)C(C)CC)NCC1(C(=O)NCC2CC(O)C2(C)C)CC(=C)C1 C(=O)(C1=C(Cl)CC1)NCC(CO)NC(C(C)(C1(C)CC1)OC)=O C(CC(O)C(F)F)NC(c1ccn(CCNC(CC2CC(SC)C2)=O)c1)=O O=C(CCCCCCn1cc(CN2CCCCC2)nn1)N1CCC12CCC2 c1(C(=O)NC(C)CNC(C2CSCN2C)=O)cc2scc(Cl)c2[nH]1 c1(N2CCCC(CCC=C)C2)cccc(S(=O)(=O)N(C)Cc2nnnn2C)n1 c1(CNC(C(C=C)(C)CC)=O)n[nH]c2c1CN(C(=O)CC1CCC13CCC3)CC2 C1(C(=O)NC(CCNC(=O)C(=O)Nc2ncc[nH]2)C(C)C)(OC)CCCCCC1 C1(COC)CC(CNC(C2CC2F)=O)N(C(c2cn(C(C)C)nn2)=O)C1 c1(C(=O)NC2C(C(=O)NC3(C(N(OC)C)=O)CC3)CCC2)ccnc(Br)c1F c1(N(C)C)cncc(NC(C2COCCN2C(=O)Cn2nccn2)=O)c1 N1(C(Cn2cc(CNC(COC)=O)nn2)=O)CCC(CO)CC1.C1CCC(O)CC1 S(=O)(=O)(CC(=O)NCCc1ccc(CNC(c2cncn2C(C)C)=O)cc1)NC c1(N2CC(NC(c3ccc(N4CCCC4)nc3)=O)C3(C2)CC3)ncnc2c1CCCC2 C(CC(=O)Nc1ccccc1O)(C(C)C)NC(CCCCOC)=O CCCCCCc1ccc(C(CC2CC2)N(CC(=O)NC2CCOC2)C)s1.CCO CCCCCCC(C)CC(=O)N1CC2CC2(NC(c2ccc3nonc3c2)=O)C1 N1(C(c2cc(C)c(Br)o2)=O)CCCOC(CNC(C2(C)COC2)=O)C1 c1(C(N2CCC3(C2)CN(C(C2CCCO2)=O)C3)=O)cc(F)cc(Br)c1Cl C1(C(N2CC(SCC)C2)=O)CC(C)(C)CCN1C(c1cc(C)co1)=O CCC(C(=O)OC)C(=O)NC(CC)CCC(=O)NCC1(OC)CCC(C)C1 n1(CC)cc(C(F)(F)C(=O)NC(C)C(C)NC(=O)C(C)COC(C)=O)cn1 c1(CCC(=O)NCC2CCCCN2C(C2CCCC(F)C2)=O)ccc(F)nc1 C(C(CC(C)C)C(=O)NC1CC1CCOC)NC(CC(CC)C1CC1)=O C=CC1CN(C(c2occc2COC)=O)CC1NC(=O)CC1CCSC1 Cc1nc(C(=O)NC2(CNC(=O)CC3C=CS(=O)(=O)C3)CCCC2)c(C)o1 c1(C)ccc(CN(C(=S)NC(C)C(C)C)OCC)cc1 C1(CN(C(c2n(CC#C)ccc2)=O)C)CN(C(=O)C(C)CSC)CCO1 C1(C(=O)Nc2ccsc2)CC12CCN(Cc1ccccn1)C2 C1(NC(c2c(CC)nc[nH]2)=O)CCCCN(C(C2CCCS2)=O)C1 c1(CC)nc(C)[nH]c1C(=O)NCC1(F)CCN(C(c2ccoc2C2CC2)=O)C1 N1(C(=O)Nc2ccn(Cc3ccccc3)c(=O)c2)CCC2(COC(COCCO)C2)C1 CN1C2CCC1CC(CC(=O)NCC1CN(C(=O)CC3CC4(CCC4)CO3)C1)C2 CS(=O)(=NC(=O)c1ccc(Cl)o1)c1cnn2c1CN(C(=O)CC=C(Cl)Cl)CC2 Cc1cc(=NC(=O)CNC(c2ccc(O)c(CO)c2)=O)[nH]o1.C1C=CCN1 C(CC(F)(F)F)N(C)C(c1c[nH]nc1CCNC(=O)C=CC(C)(C)C)=O C(=O)(C(CC(C)C)C(C)C)NC(CC=C)CNC(=O)C(=CC1CCCC1)C C1(CNC(C(CC)OCC)=O)CN(C(=O)CC2C(=O)N(C)N=C2C)CCC1(F)F N1(C(c2cc(C)c(C)s2)=O)CCC(NC(=O)Cc2cnn(C(C)C)c2)C(C)C1 N1(C(C(C)(C)C2CCCC2)=O)CCC2CN(C(=O)CC3CC3C(F)(F)F)C2C1 N1(C(C2C(=C)C2)=O)CCCN(C(c2sc(Cl)cc2Cl)=O)CC1 C(=O)(C1=CC2C=CC(C1)C2)NCC1(O)CN(C(c2n(C)ncc2C(F)(F)F)=O)C1 c1(OCC(=O)NC(CC)CNC(c2ccoc2C)=O)ccc(C#N)cc1Cl N1(C(C(COC)N(C)C)=O)CCC2OCCN(C(c3ccc([N+](=O)[O-])o3)=O)C2C1 N1(c2c(OC)nccc2)CCC(F)(C#N)C1 C12(NC(C=CCOCCOC)=O)COC(CNC(=O)CC3CCNC3=O)(C1)C2 C1(C(=O)OC)CCN(N2CC(O)(C)C2(CC)C(=O)OC)C1(C)C C=CC1CN(C(=O)C(=O)NCCC)CCO1.C1CC(C)(C)CN1 C#Cc1cnn(C)c1C(=O)NC(C)C(=O)N(C)CCn1cnnc1 C1(NC(Cc2c(C(=O)OC)cccc2)=O)CCN(C(=O)C2=NOCC2)C(C)C1 C(=O)(CCC(=O)NCCn1cc(C2CN(CC3CC3C(=O)OC)C2)nn1)NC C(=O)(CCC1=CCCCC1)N1CCC(=CCNC(c2csc(CO)n2)=O)CC1 N1(C(=O)OC(C)(C)C)CC(CCNCCCO)OC(C)C1.c1ccncc1 Cc1cc(C)c(C(=O)NC(C2CCN(C(=O)C(C)n3cccn3)CC2)C)c(O)n1 c1(C(=O)NCCCOCCn2cc(CN(C)C)nn2)noc2c1CC(C)CC2 c1(C(N2C(C3(NC(C=CC=CC)=O)CC3)CCC2)=O)cc2ncccn2n1 c1(CN(CC)CC)cc(C)cnc1O.N1(C(CNCC)=O)CC2C(C1)O2.C1CO1 C1(CC#C)(NC(=O)Cc2ccsc2)CCN(C(=O)C(O)COC)C1 c1(CNC(C2(C3CNC3)CCCC2)=O)cnn2c1C(=O)NCC2 c1(CCCC(=O)NCC2CC(NC(=O)Cc3cnoc3)C2)nc2ccccc2s1 C1(N(C(CCC2C(C)C2)=O)C2CCC2)CCN(C(=O)CCCC(C)=O)CCC1CO C(c1cccc(CN(C)C)c1)=CC(=O)NCC(C)CNC(c1coc(CO)c1)=O C12C3CC4C(C3NC1=O)C24.C(=O)(C(C(C)CC)OC)N1CCC(CC)CC1 N1(c2ccnc(NCC3(C)CCOCC3)n2)CCC2(CNC(=O)O2)C1 S(=O)(=O)(c1cc2cc(Cl)ccc2o1)N(C)C(C1CCOCC1)=O CC(C(=O)NC1C2CC1N(C(=O)C#CC(C)(C)O)C2)C(F)(F)F c1(C(N2C(C(=O)NCC3OCCO3)CC3(CC3)C2)=O)nc(Cl)ccc1F c1(C(=O)Nc2c(CC)occ2)cc(-c2ccc(COC)nc2)c2cn[nH]c2c1 N1(C(c2c(C)nc[nH]2)=O)CCCC(C2CCN(C(=O)Cc3cnns3)CC2)CC1 c1(C(=O)NC2(C3N(C(c4c(C)cns4)=O)CCC3)CC2)cccc(Br)c1C C1(C(=O)NCCCN(C(c2c(C)nc(C(C)OC)s2)=O)CC)CCC(C)(C)CC1 N1(C(CC2(NC(C)=O)CC2)=O)CC2CCCN(C(C3CCCOC3)=O)C2C1 C1(C(N(CCCO)CC#C)=O)CCCN(C(c2cccc(CO)c2)=O)CC1 c1(C(N2CC(C)C(CCNC(=O)C(C)S(N)(=O)=O)C2)=O)cnn2c1OCCC2 Cc1cc(C(=O)N(CCCC(=O)NC2CN(C)CC2(F)F)C)ncc1F c1(C(=O)OC)cnc(N(C2CCN(C(=O)CC34CCCC3C4)C2)C)c(C)c1 c1(NC(=O)NCC2CC(n3cncn3)C2)ccc2c(c1)CCC2 c1(C(N2CCC(N(C(C3CCC3)=O)CCO)C2)=O)ccnc(Cl)c1O.O=C(CN)OC Cc1nn2ncccc2c1C(=O)NCC1C2CN(C(C3CC(F)C(=O)N3)=O)CC12 c1(CC(=O)NC2(C(N(CC(C)(C)OC)C)=O)CSC2)cccnc1C N1(C(c2c(C)cnnc2)=O)CCC(C(=O)Nc2ncccc2Cl)C(O)C1 CC1(C)CC(COC(c2cnc3n2CCCC3)=O)NC(=O)N1 Cc1nn(CC(F)F)cc1C(=O)NCC1(F)CC(NC(=O)C(C)CN(C)C)C1 N1(C(C(C)c2ccco2)=O)CC2CC(C1)N2C(C1CCCCCS1=O)=O C=CCC(C)C(=O)NC1(CNC(c2ccc(NC)cn2)=O)CC(OC)C1 S(=O)(=O)(c1cc(C)cc(Br)c1)NC1CC(Nc2cc(SC)ncn2)C1 C=CC1(NC(=O)CC2(C)CCN2C(=O)Cc2sccc2C)CCOCC1 N1(C(CCCN(C(CC(C)C2CC2)=O)C)=O)CCC(C2CCOC2)C1 C1(NC(=O)COCC(F)F)CC2(C1)CN(C(=O)CN1CCSCC1)C2 N1(C(C(C)OCC)=O)CC2CC2(C(=O)N(CC(O)CO)C(C)C)C1 C1(NC(CC=C)=O)CCN(C(c2cncc(NS(C)(=O)=O)c2)=O)CC1(C)C c1(C(=O)NCC2C(C(N(C(CC(C)C)C)C)=O)CCO2)cnccc1C#N C(=O)(C(O)CCC(C)C)NC1C(CNC(CCCCSC)=O)CCCC1 N1(C(C(CCC)C)=O)CCS(=O)(=O)C(CCNC(=O)CC(F)(F)C(F)F)C1 C1(NC(c2cnn(CCF)c2)=O)CC2(C1)CN(C(=O)C(C1CCCO1)C1CC1)C2 c1(NC(c2nccc3cc[nH]c23)=O)c(Cl)cc(F)cc1[N+](=O)[O-] C=C1CC(NC(=O)NCCN2CCCCC2)N(C(=O)OC(C)(C)C)C1 C(C1CCCCCC1)=CC(=O)NCC1CC(C(C)(C)C)N(C(C23CCC2C3)=O)C1 Cc1cc(C(=O)NC2CCC(C)(CNC(=O)C3=COCC3)C2)cc(C)c1Cl N1(C(c2cncc(C#C)c2)=O)CC2CC(NC(=O)COc3ccsn3)CC2C1 Cc1ncc(Br)c(C(=O)NCCCNC(=O)C(n2cc(Cl)cn2)C)n1 C12C3CCC(C3)C1NC2=O.C1(OCCOCC)CN(C(C2CC23CC3)=O)C1 CN1CC(NC(=O)C(c2ccccc2)NC(c2ncc(F)cn2)=O)CC1=O N1(c2cc(OC)cc(C(N)=O)c2Cl)c2ccccc2NC(=O)C1(C)C C1(C(=O)NCCOC(C)(C)CNC(C2CC(O)CN2C)=O)(OC)CCCOC1 c1(C(=O)NCn2cc(CCSCC(N)=O)nn2)ccccc1Cc1ccno1 c1(CC(C(=O)NCCCN(C(C(CC)OCC)=O)C2CC2)C)cccc(C)c1 N1(CCC(N2CC(C)C(CNC(C3CC3F)=O)C2)=O)Cc2ccccc2C1 CN1C(=O)CCC1C(=O)NCC1(CNC(c2c[nH]cc2C2CC2)=O)CC1(F)F C1(CNC(C(CSC)C)=O)CCCCCN1C(=O)Cc1cc(C)no1 c1(C(=O)NCCCN(C2CCCC2)C(c2cncs2)=O)cc(Cl)c(F)cc1Cl CC(C(=O)NC1CC(CCC(=O)NC2CCCC2C#N)C1)S(N)(=O)=O C1(NC(C2CC3CCC2CC3)=O)CCCN(C(=O)C(F)CC2CC2)CC1 N1(C(c2c[nH]c3nccc-3c2)=O)CCC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 c1(C(=O)NCC2CCN(C(C(C(=C)Cl)(C)C)=O)CC2C)ccn2nncc2c1 c1(C(=O)NCC(C)CNC(c2cncn2C2CC2)=O)cccc2cnnn12 C1(C)(C(N2CC(C(C)NC(c3cc(OC)n[nH]3)=O)C2)=O)COC(C)CO1 C1(CNC(C2(OC)CCCC2)=O)CCN(C(=O)Cc2c(C)nn(C)c2C)C12CC2 C1(c2ccno2)(C(=O)NCC(C)NC(C2CCCO2)=O)CCOCC1 C1(C(=O)Nc2cccc(C(C)O)c2)CC12CCN(Cc1nc(Cl)ccc1Cl)C2 C12(CNC(c3cccc(C(F)F)n3)=O)CCCC1CN(C(C1CCC=CO1)=O)C2 C1(C(=O)N(C2CC2)Cc2cccc(O)c2)(OC)CCN(C2CCOC(C)C2)CC1 Cc1nonc1C(c1nnnn1CCC1(C)CC1)NCCCCCF N1(C(C(C)=CC)=O)CCC2(CC1)C(OC)CC2NC(=O)C1=CCSC1 N1(C(CCC=CC)=O)CC2CC(C1)N2C(c1ccc(C2CC2)o1)=O c1(CNC(C(=O)NC2C(CN(C)C)CCC2)=O)nc2c(s1)CC(C)(C)CC2 C1(C(C#C)C)CCN(C(=O)CNC(=O)CNC(C2(C)CCCO2)=O)CC1 C(=O)(C(CC(C)C)OC)NC(C1(C(=O)NC(c2ccnn2C)CC)CC1)C C(=O)(C(F)CC(C)(C)NC(=O)CCSCC)NCC(CCC)C c1(CC)cc2c(N(C(=O)C(C)CCNC)CC(C)O)nc(C)nc2s1 O(NC(=O)C(C)(C)C(C)NC(=O)C(C)S(N)(=O)=O)CC(C)O CC1(C(=O)NC23CC2CN(C(c2nnn(C(C)(C)C)n2)=O)C3)CC2(CCC2)C1 C(=O)(CCCCCCCC)N1CCN(C(CC=C=C)=O)C(COC)C1 C#Cc1ccc(C(=O)N(CC(O)CNC(C2CC(CC(C)(C)C)C2)=O)C)cc1Cl C12CC3CCC(C1)N3C2=O.C1(CNC(C2CC2F)=O)(CSC2CCC2)CC1 C(=O)(C(CO)OCC1CCCC1)NC(CNC(C=CC=CCC)=O)C1CCC1 N1(C(C=CC(C)C)=O)CC2CN(C(c3cc(F)c(Br)cc3Cl)=O)CC2C1 CCCC(C(=O)N1CC2(CCCN(C(c3c(Cl)cnn3C)=O)C2)C1)S(N)(=O)=O Cc1nc(N2CCCCC2CNC(=O)C(C2CCOCC2)F)c(F)c(C)n1 c1(C(C)C)ccc(S(=O)(=O)N2CCN(C)CC2)c(Cl)c1.N1CCCC1C(=O)CNC=O C1(NC(CN(C)C(C2CCCCC2(C)C)=O)=O)CC12CCCCC2 C1(CNC(C2OCC(C)C2)=O)CCN(C(=O)Cc2cnccn2)CC1 N1(C(=O)COCP(C)(C)=O)CC(O)CC1CNC=O.Cc1nc(CCC=O)cs1 CC(C)(CC(=O)NCC(C)(C)C#CC(=O)NCCc1ncc[nH]1)C(F)F C1(NC(c2ccc(C)o2)=O)CC(C)CN(C(C2CN(CC(C)C)C2)=O)C1 CCCCCCCCC(C)CC(=O)NCCCCNC(=O)CCn1ccnc1C C1(CC(=O)NCC(CNC(Cn2c(C)ccc2C)=O)O)CCC(C)(C)CC1 C1(C(N2CC(n3cc(-c4nc(Cl)cs4)nn3)C2)=O)CC(=O)N(O)C1 c1(CNC(c2nccc(OC)c2F)=O)ncc2ncn(C)c2n1 C1(NC(c2cc[nH]n2)=O)CN(C(c2cn3c(n2)CCC3)=O)C2(CCC2)C1 N1(C(CC(C)N(C)C(c2sccc2CO)=O)=O)CCC2(C1)CN(C)C2 Cc1ccc(=O)n(CC(N2CCC(C)C(NC(C3CC(C4CC4)=NO3)=O)C2)=O)n1 C(C(CCO)C(F)(F)F)NC(=O)NCCCCc1ccccc1 Cc1ccc(S(=O)CCNC(=O)C(c2ccc(F)cc2)c2ccccc2)cc1 c1(CC(=O)NC(CCCC)CNC(=O)C(C)(C)C2CCCO2)cccc(Cl)c1Cl N1(C(CN2CC(=O)NCC2)=O)CC(CNC(C2(CCO)CC2)=O)N2CCC1C2 N1(C(C2C(C=C)CC2)=O)CCCC(C)(CNC(c2ocnc2C2CC2)=O)C1 Cc1ccc(N2CC(C(=O)NCc3ccc(C4OCCO4)cc3)C2)nc1 C(N=c1[nH]c(C(N2CCC(N3CCOCC3)C2)=O)cs1)c1c(C)cco1 C1(C(=O)NCC(CNC(C(CC)n2cncn2)=O)(C)F)C2CCCOC12 C(CC(C)(C)CC(=O)N1CC2CCC(Nc3cc(OC)ncn3)(C2)C1)OC C(=O)(CC(O)C(C)CC)NCCCOCCC(=O)NC(CC=C)CC(=O)OC Cc1cc(O)c(C(=O)NCC2CN(Cc3c(F)cncc3F)C2)cc1Br Nc1cccc(Cl)c1C(N1CC(N2CCCC2)C(F)C1)=O c1(C(N2CC3(CCN(C(C(C(C)(C)C)=O)=O)C3)C2)=O)nc(Br)n2ccccc12 n1(CC)cnc2c(NCCC3CC3(Cl)Cl)nc(N3CCCCC4(CCC4)C3)nc12 N1(C(CCSCC)=O)CCC(NC(=O)CN2CCCC(CC)C2)C(F)C1 C12(NC(c3c(C)oc(C(C)C)n3)=O)CCCC1CN(C(=O)C(C)N(C)C)C2 c1(CC)ncccc1C(=O)NC1CCC1C(N1CCC(CN2CCCC2)C1)=O c1(COC(C2CCC(OC)CC2)=O)c(O)ccc2c1CCC2 N1(C(COC)=O)C2CCC1CN(C(c1ccc(-c3nnc(O)o3)cc1)=O)CC2 c1(C(N2CC3(CCN(C(c4ccns4)=O)C3)C2)=O)nc2n(c1Cl)CCCC2 C1(CONC(Cn2cc(C=C(C)C)nn2)=O)CC2CC1CC2O C1(C(N(CC(C)N(C(Cc2c(C)n[nH]c2)=O)C)C)=O)CCc2cc(F)ccc2O1 C1(NC(c2ccc(CN(C)CC)cc2)=O)CCCCC(O)CNCC1 Cc1cc(Br)cc(N)c1C(=O)NC1CC1CNC(=O)CN1CC2CC2C1 C(=O)(CN=S(C)(C)=O)N1CC(CC(C)N(C(c2nc(C(C)C)oc2)=O)C2CC2)C1 N1(C(c2ccc(COC)cc2)=O)CCCCC(CNC(=O)C(C)(C)C(C)O)C1 C1(C)(C(N2CC(n3cc(-c4ccc(C)nc4)nn3)C2)=O)CCCCC1C Cc1nc(N(C)C)cc(N2CCN(CC3(CC(C)C)CCCC3)C(C(C)C)C2)n1 C(CC(C(C)C)NC(C1CC1c1ccc(F)cc1)=O)N(C(C1C(C)=CCS1)=O)C C1(C(=O)NC(C2CCCC2)C)CCCN(CC=Cc2ccccc2)C1 C1(NC(Cc2cn(CC)nc2)=O)CN(C(C2CCC2)=O)C2CCCC12 C1(C(=O)NCCC(C)SC)CC(NC(=O)CN(C)C(N)=O)C(O)C1 C1(NC(CC2(OC)CC2)=O)COCC1CNC(=O)Cc1occc1C C1(Nc2nc(C)nc(=N)[nH]2)CC2(CCN(C(c3ccc(CC)cc3)=O)CC2)C1 C1(NC(C(=O)NCC(C(F)(F)F)OCCCC)=O)CN(CCOCC)CCCO1 C=C(C)CCC(C)N(C(=O)CCCC1CCN(C(=O)C(C)(Br)Br)CC1)CC c1(NC(C2C(CN3C(CCOC)CCC3)C2)=O)cnn(C)c1Br C1(NC(c2sc(C)c(O)n2)=O)CCN(c2ccc(C(F)(F)F)nn2)CC1(C)C c1(NC(=O)NCCCS(=O)(=O)NC(C)C)nc2cc(F)ccc2n(C)c1=O c1(C(=O)NCC(CNC(C(C)c2ccsc2)=O)F)scnc1C1CC1 c1(C(N(CCC)CCNC(=O)C(CC)N(C)C)=O)cnc2c(c1)COCC2 N1(C(c2cn(C)nc2)=O)CC(NC(=O)Cn2cnnn2)C2CC12 Cc1cn(C(C)C)cc1C(N1CC(O)(CO)C1)=O.C(CO)NCCN(C)C(C)C c1(OC)ccc(C(N2CC3CC3(CNC(C3OCC3(C)C)=O)C2)=O)c(Cl)n1 c1(C(=O)NC2C(CNC(CC(C)C(F)F)=O)C2)cc(=O)c2ccccc2n1C c1(CN2CC(F)CC(C(N(CCC)CCC)=O)C2)ccc(F)c2ccoc12 N1(C(CCCCN(C)C)=O)CC2CC1CCC2NC(c1coc(CC2CC2)n1)=O n1(CC)cc2ccc(C(=O)N(CC(O)CN(C(=O)CC(C)(C)C)C)C)cc2n1 c1(C(=O)NCCN(CCC)C(C2CC(F)C2)=O)ccnc(OCCO)c1 C1(CNC(c2cc(COC)no2)=O)CN(C(=O)C(C)CC2CCC2)CC1C C1(CC)(NC(c2cc(C)n(C3CC3)n2)=O)CCCN(C(=O)CC2(C)CC2)C1 N1(C(C2CC(CC)C2)=O)CCN(C(c2cc(Br)sc2C)=O)CC1C N1(C(c2cc(C)no2)=O)CCC(C(C)(C)CNC(C2(CO)CCCO2)=O)CC1 C(C(C)(O)CC(=O)NC(C(=O)N(C)Cc1ccncn1)C1CCCO1)OC CCCC1C(=O)N1.c1(CSCC(=O)OC(C)C)cnc(C)nc1 c1(COC)cccc(N2CCOCC2)c1.C1(=O)C(N(CCC(C)C)C2CC2)CN1 N1(C(C2CCC(C)N2C(=O)CC2=NN(C)C(=O)C2)=O)CCC2(CC1)CN(C)C2 N1(C(=O)OCCOC(CC)(C)C)C(=O)NC2(CCCS(=O)(=O)CC2)C1=O.N1(C)CC1 c1(C(=O)NC(c2nocc2C(=O)NCCn2cnnn2)C)cc(=O)cc[nH]1 c1(C(=O)NC2CCCCN(C(C(C)C3CCOC3)=O)C2)nc2cccnc2s1 CC1(F)COCCN(Cn2cc(-c3cccc4c3OCCO4)nn2)C1 C1(N(C(c2cnc(C)o2)=O)C)CCN(C(=O)C2CC2)CC1.CCO c1(OC)c(O)cc(C(=O)N(C2CCN(C(=O)C(C)n3ccnc3)C2)C)cc1C#N c1(CNC(=O)CNC(=O)NCc2nccs2)cnccn1 c1(OC)ccc(F)c(C(=O)NCC2C(C)CCN2C(C2CCCN2C)=O)c1 S(=O)(=O)(c1cccs1)NCC(N1CCC(O)(Cn2cc(-c3ccco3)nn2)C1)=O N1(C(c2c(OC)nn(C)c2)=O)CCN(C(C2(F)CC2C)=O)CC1c1cnn(C)c1 N1(C(COCC(=O)OC)=O)CC(NC(=O)Nc2ccc(C(C)(F)F)nc2)C2CC12 C#CC1(C)CCCN(C(=O)CC2CCCN(C(=O)CCC(C)(C)OC)C2)C1 Cc1ccc(-c2nc(C3CCCC3)nn2C)c(C(F)(F)F)c1 CCC(C)C(O)CNC(=O)CCCNC(C1(CC(C)C)CCC1)=O c1(C(N(CC(=O)N(CCC#C)C)CC2CC2)=O)nccnc1OC C1(CNC(c2csnc2Br)=O)CCCC(CNC(=O)CCC2CC2)C1 C1(C)(C(=O)NC2CN(C(c3c(CC)occ3C)=O)CC2F)CC(C2CC2)=NO1 Cc1ccc(S(=O)(=O)N2CCN(C3CCOC3)CC2)cc1C#N Cc1nccc(Br)c1N(C(C1CC(=O)OC1(C)C)=O)C1CC1 N1(C(C(CC)C)=O)CC2CCC(C1)N2C(c1cnn(-c2cccc(F)c2)c1C)=O C(C)(CC(C)N=c1nc(C(C)(C)C)[nH]s1)NC(C(CC(C)C)NS(C)(=O)=O)=O N1(C(COC)=O)CC2CCCCC2(Nc2ncnc(C)c2F)C1 N1(C(CCOCCC)=O)CCC(C)CC1C(N1CCN(C(=O)NC)CC1)=O CCCCC(O)C(C)C(=O)NC(CC(=O)NCC(C)(CC)OC)C(F)F N1(C(CC(C=C)(C)C)=O)CCC(C2CC(NC(c3cnc(OC)c(Cl)c3)=O)C2)C1 C1(C(C(=O)NCC2CC(C(=O)NCC3CCCCO3)C2)F)CCCCC1 N1(c2n(CCCC3(C)CC3)c(-c3cc[nH]n3)nn2)CCC2C(C1)C2(F)F c1(C(C(=O)NCC=C)NCC(=C)Cl)cccc(CCC=O)c1.C(CCF)OC(C)(C)C c1(CCC(=O)N(C2CCN(C(=O)CN(C)C(N)=O)C2)CC)cc2ccccc2s1 C1(F)(CNC(c2cnn(C3CCCC3)c2)=O)CN(C(c2cnc(O)s2)=O)C1 C1(CNC(CN2C(C)CC2)=O)CC12CCN(C(=O)COc1ccsn1)CC2 c1(C(=O)NCC(CC(C)C)NC(=O)C(F)C(F)(F)F)cc2c(cc1Cl)CCCC2 CC(C)CC(C(=O)NC1CCCC1NC(=O)Cc1cccs1)C(C)C c1(C(=O)NCC(CC=C)NC(=O)CC2CC23CC3)c(C)ccc(C)c1N C12(NC(C(=Cc3ccco3)C)=O)CCCC1CN(C(=O)Cc1coc(C)n1)C2 CC(CC(=O)N1CC(NC(=O)CCCCN2CCCCC2)CC(O)C1)C(F)F N1(C(CCN(CC)CC)=O)CCN(C(=O)CCCc2ccccc2)C2CC12 C1(CNC(c2c(CC)scn2)=O)CN(C(=O)CN2CCN(C3CC3)C2=O)CCO1 N1(C(c2cn(CC)nc2)=O)CC(CNC(C2CC(OC)C2)=O)CCC1C c1(CC(=O)NCC2CCCN2C(=O)C#CC2CCCC2)c[nH]c2cccc(Cl)c12 Cc1nc(N(C(=O)C(CC(F)F)C2C(OC(F)(F)F)CNC2)CCl)ccc1C(F)F C(CCC(C(=O)NN1CCCC1C(=O)NCc1cccc(O)c1)NC(C)=O)OC Cc1cnc(NC(=O)CC2CCCCN2Cc2ccc(Cl)s2)c(Cl)c1 C(CCN=C(NCc1nccs1)NCC1CC1C(C)C)(C1CCOCC1)OCC C(=O)(C(Cc1cc[nH]n1)NC(=O)CSCCC#N)N(CC(C)C#N)C c1(C(N(c2ccccc2)C(C)=O)=O)cnc(NCCC2CC2)cc1C c1(C(=O)NCCC(CC)(C)NC(c2ncnc(C)c2C)=O)ccc2nc[nH]c2n1 c1(C(=O)NC2CCN(CC)C2)cc(-c2nn[nH]n2)cc(O)c1 C1(C(=O)NCC=CCNC(C(C)NC(c2ccoc2)=O)=O)CC2CCC2C1 C=C1Cn2c(C(=O)NCC3CC(NC(c4cc(C)[nH]c4C)=O)CC3O)nnc2S1 c1(C(N(CCC(=O)N(CCC#C)C)C)=O)cncc(Cl)c1 C1(NC(CC2(CS(N)(=O)=O)CC2)=O)COC2CN(C(=O)C3=CCCCC3)CC12 N1(Cc2cc(C)c(O)c(C)c2)CC(CC2CCCCN2)c2ccccc21 NC(=O)CCC(=O)NCC1C=CCN1C(=O)CCN1CCCCCC1 C1(c2cn(C)nc2)CCCCN1C(c1c(I)cnn1C)C(=O)NC1CC1 c1(C(c2nnnn2C2CC(F)(F)C2)Nc2c(C)ccs2)cc(CO)n(C)n1 N1(C(COc2ccn(C)n2)=O)CC2C=CC1C(C(N1CCOC3CC13)=O)C2 c1(NC(C2CCC(NC(=O)OCC=C(C)C)C2)C)noc2c1CCCC2.C1CO1 c1(C(=O)OC)nccnc1C(=O)N(CC(O)CN(C)C(c1ccc(O)nn1)=O)C C(=O)(CCC(C)(C)C)N(C1CCCN(C(C2CC(=O)N(C(C)C)C2)=O)CC1)C N1(C(CCC2CC(NC(c3ncn(CC)n3)=O)C2)=O)CCC(F)(F)CC1C c1(NC(c2ccc(N(C)C)nc2)=O)cc2ccccc2nc1F C1(CC(=O)NCC2(CC)CCCC2)CCCCN(C(=O)COC(C)C)C1 Cc1ccncc1CC(=O)N(CC(=O)NC(C)(C)C)C Cc1cc(Cl)cc(C)c1OCC(=O)NC1CC(CNC(=O)C2CC2)C(O)C1 N1(Cc2cc(C)cc(O)c2)CCC(F)(F)C(C(=O)NCc2ccnc(C)c2)C1 c1(C(C(=O)NC(CC)(C)C)N(C)CCN(c2ccccc2)CC)ccc(C)nn1 CC(C)C(C(=O)N1CCN(C(c2ccc[nH]2)=O)CC1c1ccnn1C)C(C)C Cc1c(C(=O)NCc2ccnc(C(=O)NCC(=O)N(C)C3CC3)c2)cncc1F c1(C(=O)NC2CN(C(C(C)OCc3ccccn3)=O)C2)cn(C)nc1C(C)(C)C C1(C(C)C)CN(CCCc2coc(C3CCOCC3)n2)CCO1 N1(C(C(=Cc2ccco2)C)=O)CC2CCC1C1CN(C(=O)C#CC(C)(C)C)CC21 c1(CC)c(C(N2C(C(=O)NCC(=O)NCCO)CC2C)=O)ccn1C c1(C(C)(C)OC)cn(CCNC(C2(Cl)CC2(C)C)=O)nn1 Cc1cccn2ncc(C(=O)NC(C)(CNC(c3cnc(C)n3C)=O)CO)c12 c1(CC(C)C(=O)N2CC(O)(CNC(C3CCSC3)=O)C2)cccc(C(F)(F)F)c1 c1(C(=O)N(C2CCCC2F)c2ccccc2)cnc(C2CC2)nc1 N1(C(c2nc(C)[nH]n2)=O)CCOC(CCCNC(c2c[nH]c(C(N)=O)c2)=O)C1 C(=O)(CCC(F)(F)C(F)(F)F)NC1CC(C(=O)NC2C(C)(C)CC(=O)NC2)C1 c1(C(=O)NCCCNC(C2(C)CCN(C)C2=O)=O)ccc(C#N)c(F)c1 N12CC(CCC1C)CNC(=O)C2NC(=O)NC.CCC(C)(C)OCC(=O)SC c1(C(C)C)cc(C(=O)N(C)CCNC(C2COC(=O)C2)=O)c(C(C)C)o1 C(=O)(CCCCC(=O)N1CCN(C(=O)CN2CCC2C)CC(C)C1)OC Cc1scnc1C(=O)N(CC(O)CN(C(=O)CC1CC1C(F)(F)F)C)C Cc1noc(C(=O)N(CCCNC(C2CC2F)=O)Cc2ccccc2)c1C C(=O)(C(CNC(C1(O)CCOCC1)=O)CC1CC1)NC(c1n(C)cnc1)CO c1(C(=O)NC(C)(C)CNC(C2(CC3CC3)CCCO2)=O)cc(Cl)cnc1O CC1CC(N=c2nc(O)c3cnn(C)c3[nH]2)CN1C(=O)CCC(F)F c1(C(=O)NC(CN(C(=O)CC2C=CCC2)CC)C)cc(C(=O)C(C)C)c[nH]1 C1(OC)CN(CC2CCCC2)CC1NC(c1ccc(-c2noc(SC)n2)cc1)=O C1(O)(CN(C(=O)C(C)(C)N2CCCCC2)C)CCCN(C(C2CC2Br)=O)C1 CCC(C)CCCCC(=O)NCC1(C)CC(OC)CN1C(=O)C(C)NC=O C=C(F)C1(CC(=O)NCCC(C)N(C)C(c2ccnc(C)n2)=O)CCOCC1 C(=O)(CCCCC(=O)NC(C)CNC(c1cncc(Cl)c1Cl)=O)NC c1(C(=O)Nc2cc(-c3ccc(C#N)s3)ncc2)ccc2nonc2c1 C1(CNC(CC(C)N(C)C)=O)CN(C(=O)CC2CCCCCCC2)CC(C)(C)O1 c1(N(C)C)ccc(CSSCC(=O)N(C(c2ccccc2)C)CCO)cc1 c1(CC(=O)NCCNC(C2C(COC)CC2)=O)cc(OC)ccc1OC N1(C(C(CSC)O)=O)CC2CC2(CNC(=O)Cc2cncnc2)C1 c1(N2CCC(CCC)C2)nc(=NCCCCC(C)(F)F)nc(N2CCOCC2)[nH]1 c1(C(C(=O)NCC(n2cc(CC(CC)(C)O)nn2)C)(C)C)cccc(SC)c1 N1(C(CC=CC=C)=O)CCC(C2CCC2)(CNC(=O)C(C)O)CC1 C1(NC(=O)Cc2ccno2)CCN(C(c2coc(C3CCC3)n2)=O)CC(O)C1 c1(NC(CC2OCC(C)N(C(=O)OC(C)(C)C)C2)=O)cc(F)cc2ccncc12 C1(N(C)C(c2cc[nH]n2)=O)C2CN(C(C3(C)CC3Br)=O)CC12 c1(CNC2(c3n(CCCCCC)nnn3)CCOC2)ccc(C(C)N(C)C)cc1 C(=O)(C(F)C(CC)CC)NCC1CCN(C(C(C)OCCCC)=O)CC1O CC1(C)CCC1CC(=O)C(CO)=O.C1(CN(C(C2(O)CCC2)=O)C2CC2)CCCOC1 c1(CNC(C2CN(C(c3ncn(C)c3C(F)(F)F)=O)C2)=O)ccc(F)nc1F Cc1cccc(CNC(=O)C#CCNC(c2cccc(O)c2)=O)c1 c12ccc(cc1)NC(=O)C21CC1.N1(C(=O)C(F)C2CCC2)CC(O)(C(F)F)C1 Cn1nnc(NC(=O)CC(c2ccccc2Br)C2CC2)c1NC(=O)CC#N C(=O)(CC(C)(F)F)NCC(C)(C(C)C)NC(CCC(C)C)=O N1(C(CC(CC)N(C(=O)C(O)CSC)C)=O)CC2(CNC(=O)N2)C1 C1(C(N(CCCCO)CC)=O)CN(C(=O)CC2(O)CCC2)CC1(C)C CCC(C)(CNC(C1CCOC(C)(C)C1)=O)C(=O)NC(c1ncccn1)CC CP(C)(=O)C1CCCC=C1C(=O)N1CC(F)(CNC(=O)CN2CCSCC2)C1 C(Cc1ccc(C)cc1)(CC(=O)O)NC(C(C)NC(CC)(C)C)=O c1(C(N(CCNC(C2CC(CC)(CC)C2)=O)CCOC)=O)nc(C)n(C)n1 N1(C(C2CCN(C)C2=O)=O)CCC2CN(C(c3cc(C#N)ccc3O)=O)C2C1 c1(C(N(CCN(C(=O)C(C)N2CCC2)C(C)C)C)=O)cccc(O)c1[N+](=O)[O-] N1(C(Cc2c(C)noc2C)=O)CC(NC(=O)C2=CC(O)CCC2)C(N=[N+]=[N-])C1 C1(CNC(Cc2cccc(OCC)n2)=O)CCN(C(=O)C(C)NC(C)=O)C1(C)C N1(CCNC(c2cnc(CCCC)s2)=O)CCC(N=c2[nH]nc(COC)s2)CC1 N1(C(C(CC)OCC)=O)CCCC(CC)(NC(c2ccccc2C(C)O)=O)C1 C12(CNC(c3ccc(OC)nc3Cl)=O)CCCC1CCN2C(=O)C=CC1CCC1 C1(CNC(c2n[nH]c3c2COC3)=O)CN(C(c2ccccc2)=O)CCCO1 C1(CNC(c2n(CC)cnn2)=O)C2CCCC1N(C(=O)C(N1CCCCC1)C)C2 CC1(CNC(=O)C(F)(F)CCn2cc(CNC(=O)CO)nn2)CCCC(=O)N1 c1(C(=O)NCC2C=CC(NC(c3cnc(CC)s3)=O)C2)nc(C)c(C)nc1C C(=O)(CCN1C(=O)CCc2ccccc21)N(CCN(C(C1ON=C(C)C1)=O)C)C c1(C(=O)NC2CCN(C(CC(CC)SC)=O)CC2)cc2ccc(F)cc2s1 c1(C(=O)OCCC(CCC=C(C)C)C)ccc2c(C)cc(C)cc2c1 c1(C(=O)NC(CC)(CNC(=O)CC2CCCCN2C(C)=O)CC)ccc(N)c(O)c1 Cc1noc(C2CC2NC(=O)CNC(=O)CNC(=O)C(N)=O)n1 c1(C(=O)NC2CCOC2C(=O)NC2(CO)CC(CO)C2)cnc(O)c(F)c1 C1(C(=O)OCC)CCN(C(C23CCCCC2OCC3)=O)CC1C1CC1 c1(C(=O)NC2(C)CCN(C(c3cc(Br)no3)=O)C2)cccc(C#N)c1 c1(CC(=O)NCC2(C(=O)Nc3cn[nH]c3)CC2)ccnc(F)c1F N1(C(C(c2ccccc2)OCC)=O)C2CCCC1CC(NC(C1CC1CC)=O)C2 N1(C(C2CC(CCC)OCC2)=O)CCC2(C1)CN(C(C1CCCC1C)=O)CCO2 C(CCF)(C(=O)NCCCCN(C)C)NC(CC(C)C)=O C1(C(=O)NC2CC(NC(c3n(C)c(C#N)cc3)=O)C2)CC2CC(O)C(C1)C2 C1(NC(c2nc(CC)oc2)=O)CC2CCC(C1)N2C(C1CC1c1cccs1)=O Cc1ccc(Br)c(C(=O)N(C2CC(NC(c3sccc3C3CC3)=O)C2)C)c1 C1(CNC(=O)C=Cc2ccccc2)CCC2CN(C(C3CCSC3)=O)CC12 C1(CNC(CSCC#C)=O)Cc2ccccc2CN1C(=O)C(C)(C=C)CC C(CCC[Si](C)(C)C)NC(=O)OC(C#CC(C)OC)OC c1(C(=O)NCC2(NC(c3cc(OC)c(O)nc3)=O)CC2)cc2n(n1)CCN(C)C2 c1(N2CCCC(CSC)C2)nc(C2CC2)nc2c1CCCC2 c1(C(=O)NC2C(CNC(C3(CC=C)CC=CC3)=O)C2)cccc(Br)c1F N(C(=NCCCSC)N1CCC(c2cc(OC)ccn2)C1)CC(CCC)C N1(C(CCN(C(C(C=C)OC)=O)C)=O)CCS(=O)CC1 c1(C(N(c2c(C)cccn2)C)=O)nc2n(c1Cl)CCN(C(c1ccsc1)=O)C2 Cc1ccc(C(N2CC3(CC3)CC2C(=O)NCCCCCCN(C)C)=O)cc1C c1(OC)ccc2c(c1)CC(C(=O)NC1CC1NC(c1csc3nccn13)=O)O2 C1(C(N(CCCC(=O)NC(C#C)C(C)OC)C)=O)CC(=O)NC1(C)C C1(C(=O)NCCCNC(c2n(C)c(=O)ccc2)=O)CCN2CCOCC12 c1(NC(CN(C(c2nccc(CC)c2)=O)C2CC2)=O)cc(F)ncc1C N1(CC(=O)N(CC(CO)(CO)NC(c2c(C)ncn2C)=O)C)CCn2ccnc2C1 C1(CC)C(NC(=O)C(C)(C)C2CC2)CCN1C(c1ccnc(C(F)F)c1)=O C(=O)(C1CC=Cc2ccccc21)NCC1(N(C(C=CC(=O)OCC)=O)CC)CC1 N1(C(CNC(C2CCCCC2C(=O)NC2CC2)=O)=O)CCN(c2cnccn2)CC1 N1(C(C2N(C(C)=O)CSC2)=O)CCC(C)C(NC(=O)C=CCn2cncn2)C1C C1(OC(=O)CCn2cncn2)CCCC(c2ccccc2)C1 c1(C(N2CC(C(C)(C)O)(CNC(C3(CC#C)CCCO3)=O)C2)=O)cc(C)nn1C O(N1CCC(CC(=O)NC2CCCN(C(=O)C=CC(=O)NC3CC3)C2C)CC1)CC N1(C(C2N(C)C(=O)OC2)=O)C2CCC1CN(C(C1CC(C)(C)CO1)=O)C2 c1(C(=O)NC(CC)(C)CNC(=O)C(C)C(F)F)cc2sc(Br)cc2[nH]1 C1(CNC(CC2ON=C(C)C2)=O)C2CN(C(=O)C(CO)N(C)C)CC12 C1(CNC(C(C)Cc2cccnc2)=O)CC2(CCN(C(=O)C=C(Cl)Cl)CC2)CO1 CC(C)CCCCC(=O)N1CCCCCC1CNC(c1ccc(CO)s1)=O C1(CC(=O)NC2C(CC)C2)CCC(NC(=O)CN2CCCCCC2)CC1 CCC(O)C(C)C(=O)NCC12CCC(CC1n1cc(CN(C3CC3)CC)nn1)C2 c1(C(=O)NCC(C(C)C)NC(c2cnc(CC)[nH]2)=O)cccc(F)c1SC C(CCC(C)(C)C(=O)N1CCC(c2nc[nH]n2)C1)NC(C(C)CC(F)F)=O c1(C(=O)NC(C2OCCN(C(c3c(C)[nH]cc3)=O)C2)C)ccnc2c1ncn2C Cc1cc(C(=O)NCC2CN(C)CCN2C(=O)C#CC(C)C)ccc1Cl c1(N2CCN(C(C)=O)CC2)nc(=NC2CCN(C)C2)[nH]c2c1CC(C)CC2 CN1C(=O)OCC1C(N1CCN(C2CN(C(=O)C(C)(C)CN(C)C)C2)CC1)=O c1(C(=O)NC(CN(C(C23CCC(OC)C2CC3)=O)C)(C)C)ccc2c(c1)CCN2 c1(C(N2CC(COC)N(C(=O)C(C)O)CC2)=O)cc2c(C)cccc2o1 C1(CNC(C=CC(CC)C)=O)CN(C(C2CC(C)(C)C2)=O)C(C)(C)C1 CC1=C(C(=O)N2CC3(CCCC3)C2C(=O)NOCC2CC2)COCC1 C1(CNC(c2n(CC)nnc2)=O)CCN(C(c2ncoc2C)=O)C1(C)C CC(C)CC(CNC(c1cn(-c2cccc(Cl)c2)cn1)=O)NC(=O)C(C)N(C)C C1(CNC(C(C(C)C)O)=O)CN(C(c2cc(CCCO)on2)=O)CCC1(C)C c1(C(=O)NCC(C)(CO)NC(=O)CC2CCC=CCC2)ccc(=N)[nH]c1 C(c1ccc(C)o1)=CC(=O)NC(CC)(C)CNC(=O)C(C1CC1)SC CC1(C)CCCN(C(C2CC23CCSCC3)=O)C1CNC(c1cccnn1)=O c1(C(=O)NCC#CCNC(C2(CC#C)CC2)=O)n[nH]c2nccc(Cl)c12 c1(C(=O)NCCCN(C(Cn2nnc(C)n2)=O)C(C)C)cc(F)ccc1C(F)F C(=O)(N=c1ccn(CC(C)C)[nH]1)C1N(C(CC(C)=C(C)C)=O)CC(F)C1 c1(C(C)C)cc2c(N3CCC(O)C(C(=O)CCO)C3)ncnc2s1 c1(OC)ccc(COC2CC3COCC3C2)nc1C N1(C(C=C(CC)C)=O)CCN(C(=O)CC2(C)CCCO2)C(C)C1 C(=O)(C1=NOC(CNC(c2csc(C)c2C)=O)C1)NCCC(CCC)C1CC1 N1(C(COCC#C)=O)CCC(NC(c2ccc(OC(C)C)nc2)=O)C(C)C1 C(C)(C(CO)NC(C1CNC(=O)N1)=O)NC(C(C)c1cncs1)=O N1(C(C(F)OC)=O)CC2C(CN(C(=O)Cc3ncc(C(F)(F)F)[nH]3)C)C2C1 c1(C(=O)NCCC(C)NC(c2n(CC)cc(Cl)c2)=O)cccc(S(C)(=O)=O)c1F CCCCCCCCN(C(=O)CC(CC1CC1)NC(c1c[nH]c(=N)o1)=O)C C(CCCC(CO)NC(C1CCCN(CC(F)F)C1)=O)NC(CCCN(C)C)=O c1(OC)ccc(-c2nc(C)c(C(=O)N(C34CCCC3OCC4)C3CC3)s2)cc1OC C1(CNC(c2n(CC)c(O)nc2)=O)CN(C(=O)C(C)n2ccnc2)CC1(C)C N1(C(Cc2cc(COC)on2)=O)CCCCC(CNC(C2CCN(C)CC2)=O)C1 C1(C(=O)NCC(CC=C)NC(c2sncc2C)=O)CCCC(C)O1 Cc1nc(C(=O)NC(C2CCN(C(=O)C(C)CC3CCCCC3)CC2)C)[nH]c1C c1(C(=O)NCCOCCN(C(C2C(C)(CC)C2)=O)C)cc(C(F)F)ncn1 C1(NC(=O)C(c2ccc(Cl)s2)=O)CCCCN(CCc2ccc(F)c(F)c2)C1 C1(N(C(C(C=C=C)C)=O)C)CCCN(C(=O)C(F)=CC2CC2)CC1 C1(NC(C2CCCCC2)=O)CCS(=O)(=O)C12CN(C(c1cc(O)ncn1)=O)C2 Cc1nnn(C)c1C(N1CCC(CN(C)C(C2CC2(C)C)=O)CC1)=O CC1CN(Cc2ccc(SC(F)F)cc2)C2CCCCC2O1 C(C1=NOC2CCCC12)NC(C1(NC(CCC(CC)=O)=O)CCSC1)=O CCC(C)(C)C(C)CC(=O)N1CC(F)(F)CC1CNC(c1coc(COC)n1)=O N1(C(CNC(=O)OCC)=O)CCC(NC(C2CC3CCN2CC3)=O)C(C)C1 Cc1ccc(C(=O)NCC(CO)NC(C2CC(CC3CC3)C2)=O)cc1N C1(C(N2CCC(CCC)(CO)C2)=O)CC2CCC(C1)N2C(=O)C(=O)NOC c1(NCCS(CC)(=O)=O)ccc(S(=O)(=O)NCC(=O)OC)cc1[N+](=O)[O-] C(=O)(C(CC)CCc1ccccc1)NCCN(C(C1C(=C)CC1)=O)CCOC c1(C(=O)NCC2N(C(CCC(C)=O)=O)CCN(C)C2)cn(C)c(C)cc1=O C(=O)(CCC(C)NC(=O)C(C(C)C)N(C)C)NCCOCC#C N1(C(COC(CC)CC)=O)CC(O)(CNC(c2ncsc2C)=O)C1 c1(C(=O)NCCCCCN(C(=O)CCc2cccs2)C)ccc2oc(O)nc2c1 N1(C(c2nnc(O)o2)c2ccccc2)CCC2(CC1)CC2C(=O)NCc1onc(C)n1 c1(C(N2C(C)CCC(NC(c3c(CC)occ3)=O)C2)=O)cc(F)c(F)c(Cl)c1F N1(C(C2N(C(COCC#C)=O)CC2)=O)CC2CCCC(C1)N2C N1(C(C2CCC(=O)NC2)=O)CCC2CCCC12C(=O)NC1CCCOC12CCC2 C(c1nc2ccccc2o1)=CC(N1CC2C(NC(=O)COC3CCCC3)C2C1)=O N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(NC(=O)CCC(C)CC)C1C c1(CNC(=O)NCC(C(C)C)CNc2ncccn2)ccc(F)cc1F C1(NC(=O)CCN2CCCC2)CC2CC(NC(=O)C(F)(F)c3cnccn3)C1C2 N1(C(CS(N)(=O)=O)=O)C2CCCC1CC(NC(=O)C(F)CC1CCOC1)C2 n1(C(C)C)cc(C(=O)NC2CCC(NC(C3(CO)CC3)=O)C2)ccc1=O C(=O)(C(CC1CCC1)NC(C1(NC(=O)CC(C)C2CC2)CCCC1)=O)OC c1(C(=O)NCC2CN(C(C(COC)N(C)C)=O)CC2C)cc(C#N)ccc1F N1(C(C(CC2CCC2)OC)=O)CCOC(C(=O)NCCc2ccncn2)C1 N1(C(c2cccc(OCC)c2)C(=O)NC2CCC2)CC(CC)OC(C)(C)C1 C(=O)(CCCCCCCBr)N1CC(O)(CN(c2ccccc2Br)C(CC)=O)C1 C#CC1(C(N2CCC(C(C)CNC(=O)C(CN(C)C)N(C)C)CC2)=O)CCCC1 C#CC1CN(C(=O)C=CC2CCCN2C(c2nnsc2C)=O)CCO1 C1(NC(C(CC=C)(C)C)=O)CN(C(C2CC3CCC(C2)O3)=O)CC1N=[N+]=[N-] C12CC13CCN(CC3)CC(=O)N1CCCC(C1)N(C)C2=O.C1(NOC)CCCC1 C1(NC(C(C)OCCC(C)C)=O)CN(C(=O)C=Cc2ccccc2)CC2(CC2)C1 c1(OCC(=O)NCC)c(Cl)cc(C(=O)NC2CC2N2CCCC2)cc1Cl c1(NC2CC(CNC(c3nc[nH]n3)=O)C2)ncnc2c1ncn2C1CC1 CCC(CC(=O)N1CC2CC(NC(=O)CN3CC(C)C3)C1C2)C(C)C c1(OC)cnc(C(N2CC3C(C2)N3C(c2cccc(F)c2OC)=O)=O)c(F)c1 c1(C(N2CC(C)C(C)(CO)C2)=O)cc2cccnc2[nH]1.C12(C)CN(C1)C2=O Cn1oc(C(=O)NCC(CO)NC(c2ccc(CSCC(F)(F)F)o2)=O)cc1=O c1(N(C(=O)NC(c2c(C)nn(C)c2)C)CC)c(F)cccc1Cl.C(C)(C)C N1(C(C(CC(F)F)NC(C(C)(C)n2cnnn2)=O)=O)CC23CCC2(COC3)C1 c1(C(=O)NC2CCN(C(c3ccc(Br)c(Br)c3)=O)CC2)cnc2ccoc2c1 CC(C)C(C(=O)NC1CCC(NC(=O)CC(C)(F)F)C1)c1ccccc1 c1(OC(F)F)cc(S(N)(=O)=O)cnc1NC1COCCOC1 C1(CC)(NC(c2cccc(N)c2)=O)CCCN(C(c2cnccc2N(C)C)=O)C1 C1(CCC(N2CC(=C)C2)=O)CCN(C(c2ccncc2)=O)CC1 C1(NC(C23CC(C(=O)OC)(C2)C3)=O)CCCC(NC(=O)CCC2CCCC2)CC1.SC CCC(C)CC(=O)NCCC(C)NC(c1cnn(C(C)C)n1)=O C=CC(CC)CC(=O)NC1CN(C(=O)C=CSCC)CC1c1cncn1C c1(C(N2CC(O)(CCNC(C3CC3C(N)=O)=O)C2)=O)cc(OC(F)F)cc(Cl)c1 C(CCCCC(=O)NCCc1ccc(F)nc1)NC(C1(CC)CC(C)(C)C1)=O C1(C)(NC(C2(NC(c3n(COC)ncc3)=O)CC2C)=O)CCCC1C N1(C(C(C)(F)F)=O)CCC(CO)(CNC(=O)C(C2CCCCC2)F)CC1 c1(C(=O)NC(CCOC)CNC(C2CSC2)=O)ccc(C2CCC(=O)N2)cc1 CC1(C)C(NC(c2ccn(CCNC(=O)CC3CCSC3)c2)=O)CC1(F)F c1(OC)c[nH]c(C(=O)NC(C)CCCCNC(C2CC(OC)C2)=O)cc1=O C=CCC(CC=C)C(=O)NCCC1CCN(C(c2cc(Br)co2)=O)C(C)C1 Cc1ccc(=O)n(CC(=O)NCCN(C)C(c2scc(C)c2Br)=O)c1 N1(C(CCCCOC)=O)CC2ON=C(CNC(c3cn4c(n3)CCC4)=O)C2C1 C1(CNC(c2c(C)n[nH]c2)=O)COCCN1C(C1CCCN(C)C1)=O c1(C(c2nnnn2CSc2ccccc2)NCCF)ccnn1CC1CCOC1 C(CC(C)C)(C(=O)N1CCCC1C(C)C)N(C(CN(C1CC1)CC)=O)C C1(C(=O)NCC2OCCN(CC)C2)C2CCC(C2)N1C(=O)CCc1cnc(C)o1 c1(C(N(CCNC(C2(CC#C)CCCCC2)=O)C(C)C)=O)ccc([N+](=O)[O-])s1 C1(C(=O)NCC2(OC)CN(C(c3n(CC)ncc3)=O)C2)OCCC1(C)C CCCCC(C)CCC(=O)N1CCCC1CC(N1CC(C2=NOC(C)C2)C1)=O N1(C(CC=CCC)=O)CCN(C(c2cccs2)=O)C2CC12 C(C(CNC(C1(C)CC1)=O)S(C)(=O)=O)NC(Cc1nc(C)oc1)=O C1(CNC(C2(NC(C3CCS(=O)(=O)C3)=O)CCSC2)=O)CCC2(CC2)C1 c1(C(=O)NCCCN(C(CC)C)C)cn2c(n1)CCN(Cc1ccco1)CC2 CS(=O)(=O)CCn1cc(NC(c2nc(NC(=O)C3CC3)cs2)=O)cn1 CCC(CC(=O)NCC1CC(C)(O)C1)N(C)C(C1CCN1C(C)(C)C)=O C1(C(N(CC(CCC=C)O)C)=O)CN(C(c2ccnc(C)n2)=O)CC1(F)F CSC1=C(C(=O)N(C)CCN(C)C(c2cc(OC)ncn2)=O)CCCC1 N1(C(CCC(=O)NCC)=O)CC(NC(c2sc(CO)nc2C)=O)CC12CCOC2 N1(CCN(C(=O)Nc2cc(C3CC3)no2)C(c2n[nH]cc2Br)=O)CCCC(O)C1 C(=O)(CC1COc2cc(O)ccc21)NC(C(=O)Nc1cc(CC)c(F)cc1)C CCN=c1ccc(C(N2CC(OC)C(NC(c3nc(Cl)sc3Cl)=O)C2)=O)c[nH]1 c1(CNC(C2CCS2(=O)=O)=O)ccc(C(N2CCC(O)(CO)C2)=O)nc1 Cc1cc(C(=O)NCC2CN(C(c3ccn(C(C)C)n3)=O)C3CC23)cc(N)c1Cl C(C(=O)N(C(C)CC(=O)N(CCC(C)(C)C)C)C)(C(C)C)SCC C12(NC(=O)CCOc3cccc(F)c3)CCCC1CN(C(C1(CO)CCC1)=O)C2 c1(C(N2C(CNC(C3(C)ON=C(C)C3)=O)CCCC2)=O)noc2ccc(Cl)cc12 N1(C(CC(C)N(C)C)=O)CCN(C(=O)CCCn2ccnc2)C2CCC12 C1(C(=O)O)(CC)CCCCC1.C1(COCC#C)CCCN1C(=O)C=O C1(C(=O)NC2C(CC(=O)NCC3CCC(CC)O3)CCC2)CC2(CCC2)C1 C(C(C)(C)CC(=O)N=c1ccn(CC)[nH]1)NC(C(C=C=C)C)=O c1(CN2C3CN(C(c4ccc([N+](=O)[O-])o4)=O)CC2CC3)cc(Br)ccc1[N+](=O)[O-] c1(C(N2C(CNC(C=CC=CC)=O)CC(C)(C)C2)=O)cnc2sc(C)cn12 C1(NC(NCC(=C)C)=NCCC2CC2C(F)(F)F)CCn2c(C)cnc2C1 C1(C(=O)NC(C2CN(C(c3ccc(C(O)CF)cc3)=O)C2)C)C2CCC(F)(F)C12 c1(NC(=O)CCCCCCBr)cccc2c(C3=CCCOC3)cccc12 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(C)CNC(c1nnn(C)n1)=O c1(NC2CN(C(c3ccc(C)c(F)c3)=O)C(C)C2)ncnc2cc(C3CC3)nn12 C12(CC)CCCN(C1)C(=O)CSC(C)C(=O)N2.C(=O)(C1CC1)NC N1(C(CCN(C(c2nc(N(C)C)oc2)=O)CCO)=O)CCC(O)CC(C)C1 c1(OC)ncc(C(=O)NC(C(=O)N(C)CCn2cncn2)c2ccoc2)s1 n1(CCN(C(=O)C(=O)N(CCCN2CCCC2)C)C)cc(CCC(=O)OC)nn1 c1(NC(C2CN(Cc3ccc(F)c(Cl)c3)CCC2O)=O)cc(Br)cnc1[N+](=O)[O-] N1(C(c2nn(C)c(C(F)F)c2)=O)CCC(CO)C(NC(=O)C2=CCSC2)C1 N1(C(C2CC(=C)C2)=O)CCC(C2CC2)(CNC(=O)C(CC(C)C)NC(C)=O)C1 C1(CN(C(=O)C(F)CC2CC2)C)CCCN(C(=O)CCc2ccc(N)nc2)C1 CC1CN(C(C2Cc3cscc3C2)=O)CC(CCNC(=O)CCSCC(N)=O)O1 c1cnc2cc(CCC3(c4nnnn4CSc4ccccc4)CCC3)oc2c1 c1(C(=O)NC)ccc(C)c(NC(C)CCN(C)C(=O)OC(C)(C)C)c1 C1(NC(Cn2c(C)ccc2C)=O)CCN(C(c2ccc(=O)oc2)=O)C1(C)C N1(c2n(Cc3c(OC)ccc(OC)c3)nnn2)CCCC1C1OCCO1 N1(C(CC2C(C)(C)CCN2C(C2CCCCC(=O)N2)=O)=O)CCc2ccccc2C1 CC(C)(C)C(C(=O)NC1CN(C(c2cc(F)cnc2O)=O)CC1O)C1CCCC1 C1(C(N(C(CN(C(C(=O)Nc2ccc(C)cc2)=O)C)C)C)=O)CC(C)(C)CCN1 CN1CC(C(=O)NCC23CC(NC(=O)CN4CC5CC5C4)(CO2)C3)C(C)(C)C1 C1(NC(=O)CCC2CC2)CN(C(c2cnc(C(F)(F)F)nc2)=O)CC1F N1(C(CC(=O)OC)=O)CCC2(CCOCC2)C(NC(C2CCC3(C2)N=N3)=O)C1 C(=O)(CC(C(F)F)C(C)(C)C)NC1(C(N=c2[nH]nc(-c3c(C)occ3)s2)=O)CC1 C1(CNC(c2[nH]cc(C)c2)=O)CCN(C(=O)C(C)c2ccsn2)C(C)C1 CCCC(CCC)CC(=O)N1CCC(CF)(NC(=O)CC2CCC(=O)NC2=O)C1 C(=O)(CC(C)n1ccc(C)n1)NCCCN(C(=O)CCc1cnc(C)s1)CC N1(C(C)C(=O)NC(=O)CNC=O)CCCCC1C(=O)O.C(C)(C(O)C(F)F)N c1(-c2cccc(CC(=O)NCc3ccc(C)cc3)n2)ccc(F)c2cccnc12 C1(C(N(C(C)C(C)(C)O)C)=O)(NC(c2cn(C)cn2)=O)CC(F)(F)C1 N1(C(CCCCCC#C)=O)CC2(CCCCN(C(C3CCOC(C)(C)C3)=O)C2)C1 c1(C(=O)NC(CC)CNC(=O)CN(CC)CC2CC2)ccncc1C(F)(F)F C12=NNC(=NC(=O)NCCN1)S2.N1(SC)CCCC1 N1(C(CSC)=O)CCCC12CCN(CCNCc1nccs1)CC2 C1(C(=O)N(CCCNC(C2CC(C)=NO2)=O)CCO)(COC)C=CCC1 c1(OCC=C)ccc(S(C)(=O)=O)cc1NC(c1cnc(COC)s1)=O C1(Cn2cc(-c3ccc(C)s3)nn2)CC2CCC1N2C(c1ccn(C)n1)=O C1(C2(O)CCOCC2)(CNC(N(C)Cc2c(C)occ2)=NCc2ccccc2)CC1 N1(C(C2(C)CCC(=O)C2)=O)CCCCC(CNC(c2n[nH]c3c2CCC3)=O)C1 c1(OC)ncc(C(=O)NC2CC(CCNC(c3nccc(C(F)F)n3)=O)C2)cn1 CC(CC1CC1)C(=O)N1CCC(N(C)C)C1.C1CC(C)(C)O1 c1(C(=O)OCC)c(C)sc(C(N2CC3CC2CN3C(C)C)C(=O)NCC)c1Cl CCCC(CC)C(=O)NC(CO)CCCNC(C1CCCS1)=O c1(CC)[nH]nc(C(=O)NCC(O)CN(C(=O)C=Cc2cnc[nH]2)C)c1Cl n1(CC(=O)N(CCC(C)NC(C2(COC)C=CCC2)=O)C)cccc(C)c1=O N1(C(C(c2n(C)ncc2)O)=O)CCC2CN(C(=O)CN3CC(C)(C)C3)CCC2C1 CC(C)(CC(=O)NCC(C)(C)CNC(c1cccc(C2CC2)c1)=O)c1ccccc1 c1(C(N(CCNC(Cc2cc(CC)no2)=O)C(C)C)=O)ccc2cc[nH]c2c1F C(N1CCC2(CCCCO2)C1)c1n(CC(C)(C)C)nc(-c2cnn(CCO)c2)n1 CC1CCN(C(c2cc(C3CCC3)nn2C)=O)CC1CNC(C1(Cl)CCC1)=O S(=O)(=O)(CC(=O)NC1CN(C(=O)C(c2ccc(C)cc2)(C)C)C1)NC C1(NC(c2cncc(N(C)C)c2)=O)CCCC(NC(C2(C(C)(F)F)CC2)=O)CC1 CC1(NC(c2cnc(S)[nH]2)=O)CC(NC(=O)CSCC(N2CCCC2)C)C1 Cc1cn2cc(C(N3CC4CCN(C(=O)CC5CCN(C)CC5)C4C3)=O)sc2n1 N(C(=NC1CCCC1)NCC(C1CCOCC1)(F)F)CC(F)(F)F C(C1(C)CCOCC1)=CC(=O)NC(C1CN(C(c2ccc(CN=[N+]=[N-])o2)=O)C1)C C(N=c1cccc(S(=O)(=O)NC(C2CC3CC3C2)=O)[nH]1)C1(CC(C)C)CC1 CC(C)(C)C(CNC(C1CSCN1C(=O)CC)=O)NC(=O)Cc1ccno1 c1(C(=O)NC(C2OCCN(c3nnc(CC)o3)C2)C)cc2sccc2n1C c1(NC(C=CCNC(Cn2ccc(C)cc2=O)=O)=O)ccccc1N=[N+]=[N-] CC#CCCCC(=O)N1CCCC1C(C)NC(=O)C(C(C)C)OC c1(C(=O)NC2C3N(C(C(C)(C)N(C)C)=O)CC(CC3)C2)c[nH]c(=O)c2ccnn12 c1(C(N2CC(C)(OCC(=O)NC3(CCCC)CC3)C2)=O)c(C)ccnc1O C1(NC(C(C)(C)NC(=O)C(F)OC(F)(F)F)=O)CCCCC1C(=O)OC(C)(C)C CN1CCC(C)(C(N2CC(NC(=O)Cc3ccon3)C(n3ccnn3)C2)=O)C1 N1(C(C(C(=O)OCC)C(C)C)=O)CCCC2(NC(=O)CCC3CC3)CCCC12 c1(NC(=O)NC(c2ccc(Br)cc2)CF)ccc2oc(Cl)cc2c1 C=CCC(CC)C(=O)NC(C)CNC(=O)CC1NC(=O)NC1=O C1(NC(c2cnc(N(C)C)nc2)=O)CC2CC(C1)N(C(c1ccns1)=O)C2 C1(CN(C(c2nc(CC)oc2)=O)CC)CCN(C(C2(CC)CCCO2)=O)CC1 c1(C(N2C(C(=O)NC(C)CN(C)C)COCC2)=O)ccc(=O)n(C)c1 CC1(CNC(=O)CCOCC(F)F)CCC1NC(C12CCC(C1)C2)=O c1(C(N2CCC(F)(C(N(CC(CSC)O)C)=O)C2)=O)c[nH]c(C#N)c1C C1(CC)(NC(=O)CCOCCN(C)C)CCN(C(c2cc(Br)c(C)o2)=O)C1 N1(C(CCC(=C)Cl)=O)CC2CCC1CN(C(=O)Cc1ccccc1S(C)=O)C2 CC1CC(C)(C(=O)NC2CC(CNC(=O)CCc3cccc(F)c3)C2)CC(C)O1 CCCCC(=O)NCCC1CCN(C(c2cscc2Cl)=O)C1 N1(CC(N2CC(C(=O)NCCC3CCC(C)O3)(SC)C2)=O)CCC(O)CC1 C(=O)(C1CCOc2ccc(Cl)cc21)N1CC(C)CS(=O)(=O)CC1 c1(C(N2CC(OC)(CNC(C3CCCOC3)=O)C2)=O)cc(O)cc(N)c1C N1(C(COCC#C)=O)CCN(C(c2cccnc2)=O)CC(C)(F)C1 Cc1cc(C(=O)NCC2CN(C(=O)C(c3ccnn3C)C)CCO2)ccc1Cl Cc1ncnc(C)c1C(N1CCC(NC(C2(C)CC=CCO2)=O)C1)=O Cc1cc(C(=O)NCCN(C(=O)C(C)CC2CC2)C2CC2)ccc1-n1cnnn1 N1(C(COCCC#C)=O)CCC2(CCCCN(C(=O)C=CC(=O)NC3CC3)C2)C1 S(=O)(=O)(c1ccccc1F)N1CC(NC(c2cnc[nH]2)=O)C1 c1(C(=O)O)cc2cc(C(=O)NCCCOc3cccc(F)c3)sc2[nH]1 c1(C(=O)OC)cnc(SCC)[nH]c1=NCC1CCCN1C(=O)COCC(C)(C)C C1(OC)(CNC(c2cc[nH]c2C)=O)CCN(C(c2nncs2)=O)C1 N1(CC)CCCC(NC(=O)CC(C)(C)N(C)C(C2CC2C(N)=O)=O)C1 C(Cc1ccccc1)(CC(=O)O)NC(=O)Nc1cc(C)on1 c1(C(N(C)CCOCCNC(=O)CSC(C)(C)C)=O)cnn2c1N(C)CC2 c1(C(N2CC(OCC(=O)N(C(CC)CC)C3CC3)C2)=O)snnc1CC c1(C(=O)NCCC2CCC(NC(=O)CCc3cccs3)C2)occ2c1CCCC2 c1(C(N(CCNC(c2c(SCC)cccc2)=O)CC)=O)cc(C(C)C)ccc1F c1(C(N2C(CO)CC(NC(C(CC)(C)O)=O)C2)=O)cc(C#N)cc2ccccc12 N1(C(c2c(OC)cnnc2)=O)CCC=C(C(=O)N2CC(SC)C2)C1 C1(CC)C(NC(C2(SC)CC2)=O)CCCN1C(c1ocnc1C)=O C(C(=O)NCC1(C2CCCN2C(=O)CCOC2CC2)CC1)(C(C)(C)C)N(C)C N1(C(C(CCC)NC(c2cn(CC)nc2C)=O)=O)CCOC2(CC2)C1 N1(C(CS(CCOC)(=O)=O)=O)CCC2(CCC(NC(=O)C(CO)N(C)C)CC2)C1 C1(CSC=CC(=O)NCCNC(CCC=CC)=O)CCC(C)(c2ccccc2)C1 CC1(C)CC(CNC(c2ccc[nH]2)=O)CN(C(=O)C(c2ccc(F)c(F)c2)=O)C1 C1(C(N(CCCCC(=O)NCCN2CCC(O)C2)C)=O)CC2(C1)CC2(F)F C1(CNC(Cc2cc(C)sc2)=O)(NC(=O)COC2CCCC2)CCCCC1 n1(CC(N2CCC(CNC(C3C(C)(CC)C3)=O)CC2)=O)nnc2c1CCCC2 C1(O)(C(=O)NCC(Cc2ccccc2)NC(CC2(C)CC2)=O)CCCOC1 N1(C(CC(CCCC)O)=O)CCCC2(CCCN2C(=O)CC(Cl)Cl)C1 n1(CC(=O)OC)cc(C(N2CCC(NC(C3(C)CCCO3)=O)C2)=O)cn1 N1(C(c2ccc(C)s2)=O)CC(NC(c2cnc(C)c(C#N)c2)=O)C(C2CC2)C1 N1(N2CCC(n3cc(CCCCC(N)=O)nn3)C2)CC2CCCC2C1.C(=O)CC#N C(C(C)(C)CN=[N+]=[N-])NC(CCOCCNC(C1CN(CC)C(=O)C1)=O)=O CC1CCOC(C(N2CCOC(CCNC(=O)C(F)(F)c3cnccn3)C2)=O)C1 CC1CCC(CNC(C2CC=CC2)=O)CN1C(=O)CCc1ccccc1Cl C1(O)(CC(=O)NCC(C2CCC2)NC(c2c(COC)ccs2)=O)CCN(C)CC1 c1(NC(CCOCC=C)=O)ccccc1Cn1cc(C2CC2)nn1 C=C(Cl)CC(N)C(=O)N(O)Cc1cn(CC(CC)CC)nn1 C(=O)(CN=S(C)(C)=O)NCCCCC1(NC(C(C)C(=O)N2CCOCC2)=O)CC1 c1(CC)cnc(C(=O)NC2CCN(C(=O)CCc3nncs3)C2)nc1 Cc1ccc2c(n1)CN(C(C1CN(C(=O)CC3COC(=O)C3)CC1(C)C)=O)C2 c1(C(C(=O)NCC2C(NC(CSCCC(C)C)=O)C2)(F)F)ccc(Cl)nc1 [N-]=[N+]=NCCNC(=O)C(C1CCCC1)NC(C1CC1(F)Cl)=O C1(CN(C(=O)C(CC2CC2)NC(c2ccncc2)=O)C)CCCCCC1 c1(C(=O)NC2CC(NC(C(n3c(C)ccn3)C)=O)CC2O)cn2ccnc2cn1 C12(C3CC3)CCN(C1)C(=O)C(=O)N2.c1(OC)c(N(C)C)cccc1C(N)=O N1(C(C2C(C)C2)=O)CCN(C(C2(c3cccc(F)c3F)CCC2)=O)CC1C(C)C C12(C(=O)NC(C3(F)CCN(C(c4ccc(N)c(N)n4)=O)C3)C)C3C4C1C1C2C3C41C N1(C(c2ccc(C)c(C)c2)C(=O)Nc2ccccc2Cl)CCCCC(S(C)(=O)=O)C1 c1(C(=O)NC2CC(CNC(Cc3c(C)non3)=O)C2)ccc(C#N)nc1O C(C(C)(C)CC(=O)N(C)CCNC(=O)CC1CCN(CC(F)F)CC1)OC.O=C c1(C(N2CC(O)CC(NC(C(C(=C)Cl)(C)C)=O)C2)=O)c(Cl)cc(Cl)nc1N C(=O)(CC(C)c1ccco1)N(CCC(C)NC(c1[nH]ccc1-c1cccs1)=O)C Fc1ccc(Br)c(C(c2nnnn2C2CCOCC2)NC(CF)C2CCC2)c1 C(=O)(C1CCCc2scnc21)N(CCNC(=O)CN(C)CCOC)CC N1(C(CC(CC)(C)C)=O)CC2OCCN(C(=O)C(C)Oc3ccc(C)cc3)C2C1 Cc1nc(CN2CCN(C(=O)C(O)Cc3ccc(O)cc3)CC2CO)ccc1Br C(=O)(CC(C)CC(=O)N1CCCC(NC(C2CN(C3COC3)C2)=O)C1)OC N1(c2nnc(C3C(OCC)C3)n2CC)CC(C)c2ccc(OC(F)F)cc21 C(=O)(C1CC=Cc2ccccc21)N1C(CNC(=O)CCC2CC2)CC1 N1(C(c2n(CC)ccn2)=O)CCCC(C(=O)NCCC(C)O)C1C C12(NC(C)=O)CCC(CNC(C3CC(C)N3Cc3cc([N+](=O)[O-])c[nH]3)=O)(C1)OC2 C1(NC(CSCCCC)=O)CCN(C(=O)Cc2cncn2C)CC1CO c1(CC(CC)NC(c2ccccc2N(C)C)=O)cccc(Br)c1 c1(C(=O)NC(C)CC(C)NC(=O)CC2=NNC(=O)C2)cn(C)c2ccccc12 O=C(N=c1cc[nH][nH]1)C1c2ccccc2CN1Cc1cc(I)ccc1Br C(=O)(C1=NOC(C)(C)C1)NC(c1cn(C)nn1)C(N1CC(F)(C(=O)OC)C1)=O C(=O)(C1=CC2(CCOC2)C1)N1C(CNC(c2c(OC)cc(=O)n(C)c2)=O)CCC1 C1(C(=O)NCCOCC=C)COCCC1NC(c1csc(C)c1)=O N1(C(c2n(CC)cc(Cl)c2)=O)CC2CN(C(=O)Cn3nc(C)ccc3=O)CC2C1 C1(C(F)(F)F)(C(N2CCC(N(CCO)C(c3ccccc3S)=O)C2)=O)CCOCC1 c1(C(=O)NCC#CCNC(c2n(CC)nnc2)=O)coc2c1N(C)C(=O)CCC2 c1(OC)nc(C(=O)NC2CS(=O)(=O)CC2NC(c2ccnc(N)n2)=O)cc(O)n1 c1(OC)ccc(CSC(C)C(=O)N(CC(C)NC(=O)Cc2ccccc2)C)cc1 c1(C(CNC(=O)CC(=O)NCc2n[nH]cc2C)OCC)ccc(Cl)cc1 C=CCC(CNC(=O)CC1CC2CC2C1)C(=O)NCCNC(=O)OC C1(CC)CN(C(=O)C(C)C2CCC2)CC1NC(=O)C(C)=C(C)C C12(CCNC(c3cc(C)ns3)=O)CCC(C1)N(C(c1cc(=O)n(C)cn1)=O)C2 S(=O)(=O)(c1ccc(N2CC(C)CC(O)C2)nc1)N1CCC(N2C(NC)CCC2)CC1 c1(SCC)ccc(C(=O)NCC2(F)CCC(NC(c3cncnc3)=O)C2)cn1 c1(NC(=O)NCCN(C(=O)CC2CCC(O)C2)C)ccc(NS(C)(=O)=O)cc1O C1(CC)CCCN(C(=O)CN(C2CC2)CC)C1NC(=O)CCc1ccnn1C CONC(=O)C(=O)N(CCC(C(C)C)NC(=O)CC1CC(CF)C1)C C1(C(=O)NCCOCC)(CC)CCCN(C(C2CCOC2C)=O)C1 C12(C(=O)NCc3scc(CNC(c4n(C)ncc4Cl)=O)n3)CCOC(C)(C1)C2 C#CCC(CC#C)C(=O)N1CC2CC1CN2C(=O)CC1(CC)CCC1 C1(CNC(=O)CC2CCCC(=O)N2)CCCCN(C(=O)Cc2ccc(O)nc2)C1 C1(C(N(CC(CC)NC(C2CSCN2C)=O)C)=O)CN2CCCN1CC2 c1(C(C(=O)NCCC)N(C2CCOCC2)C)ccc(OC(F)(F)F)cc1C C#Cc1cncc(C(C(=O)N)N(CC(C)C)CCCC)c1.C(C)(C)O C(=O)(C1CCC(=O)c2cccn21)NCCC(C)NC(c1c(F)cc(F)cc1F)=O Cc1cnc(C(=O)N(C(C)CNC(c2ccc(OC(F)F)cc2)=O)C)c(F)c1 C1(NC(c2c(COC)ccs2)=O)CCN(C(=O)C#CC2(C(F)(F)F)CC2)C1(C)C CC(C)CC(C)(C)C(=O)NC1CC(NC(=O)CCC(C)N(C)C)C(O)C1 C(CNC(=O)C(=O)NCC(C)CNC(N)=O)(C(=O)NC)OCCOC C1(C(N(CCOCCNC(c2c(OC)cccn2)=O)C)=O)CCn2cnnc2C1 C1(CNC(C(=O)NCC#C)=O)CCN(C(=O)CSC2CC2)CC1 C1(CCN(C(C2CC(OC)C2)=O)C)CCCCN1C(=O)CSC(F)(F)F C1(CCC(N2CCC(OCCNC(=O)C(F)=CC3CC3)C2)=O)CCCCCC1 c1(OC)cc(C(=O)N=c2ccn(C(C)(C)C)[nH]2)cn2ncnc12 c1(C(N2CC3N(C(C=CCC)=O)C(CC3)C2)=O)cc(C)c2c(O)nc(O)nc2n1 OCCN=c1[nH]c2c(c(=NCc3cccc4c3CCCC4)[nH]1)SCC2 C1(C(=O)NC(C#C)CCC)COCCN(C(=O)CC2CCN(C)CC2)C1 N1(C(C(c2cccc(O)c2)C)=O)CCCN(C(=O)C(C)(C)C)CC1 C1(C(C)C)(C(N2CCCC2)=O)CCN(C(c2csc(F)c2)=O)C1.C1CC(C)(C)C1 N1(C(c2c(C(C)C)n[nH]c2)=O)CCC(NC(=O)C(O)CC2CCCCC2)C1(C)C C1(n2cc(CNC(C(C)OC)=O)nn2)CCN(C(C2CCS(=O)CC2)=O)CC1 c1(COC)cc(C(=O)NC(C)(CSC)CO)n[nH]1.C1(C)C=CC(=O)N1 C(C(=O)NCC1(NC(C2CC3(CSC3)C2)=O)CC1)(C(C)C)OCC C(CC(F)F)(C(=O)NCCS(C)(=N)=O)NC(C(C)(C)n1cnnn1)=O N1(C(C)Cn2cccn2)CCc2nc(C(=O)Nc3ccc(F)s3)cn2CC1 c1(NC(C(CCC)C)c2nnnn2CC2(C3CCCO3)CC2)ccc2[nH]ccc2n1 Nc1ccc(C(N2CC3CC(NC(C4CNC(=O)O4)=O)C2C3)=O)cc1F N1(C(C2CCOC3(CCC3)C2)=O)CC2(CCN(C(=O)C(F)n3cccn3)CC2)C1 CC1CCC(N(C)C(c2ccc(CNC(=O)CCc3cnn[nH]3)s2)=O)C1 c1(NC(CN(C(C2CC(O)(CC#C)C2)=O)C)C)cccc(F)c1[N+](=O)[O-] c1(CC(C)NC(N2CCC(CC(=O)OCC)C2)=O)ccc(C#N)cc1 c1(CC)ccc(C(=O)NC2CN(C(C3CC(C)OC3C)=O)C(C)(C)C2)c(N)c1 N1(C(C(C(C)O)C)=O)CCC(N=c2ccc3nnnn3[nH]2)C1 N1(C(C(CO)OC)=O)CC2(CCCC2)C1C(=O)NCC1CCOC1C N1(C(C=CC)=O)CC2CCC(CNC(C3CC34CCCc3ccccc34)=O)(C2)C1 c1(CCC(N2CC(C)(CC(=O)NCC(CC)OC)C2)=O)cn(C)nc1C CCCC(C)(CCC)C(=O)N(CC(C)(C)CNC(C1(C(=O)OC)CC(OC)C1)=O)C c1(C(N(C2CN(C(=O)C#CC(C)(C)C)C2)C)=O)cc(Br)c2occc2c1 N1(C(CC2(OC)CCCC2)=O)CC2(CCCCN2C(C2CCCC(=O)N2)=O)C1 C(=O)(CC(C)CC(=O)OC)NC(CN(C(C1CCCOC1C)=O)CC)C S(=O)(=O)(c1ccc2[nH]c(=NC3CCC(C4CC4)C3)sc2c1)NCCCC(CC)CC CC1CC(C(=O)NCC2(C)NC(=O)NC2=O)CCN1C(c1ccn(C)c1)=O c1(C(N2CCCC2CCC#N)C(=O)NC(CC)(C)C)ccn(C2CCC2)c1 N1(C(C2CCN(C(N(CCOC)C)=O)CC2)=O)CCN(CCN)CC1 C1(C(=O)NCCC(CCC)O)CC2(CCC2)CN1C(c1cccn2cncc12)=O c1(CC)cnc(C(=O)NCC2CCCN2Cc2ncccc2C(F)(F)F)nc1 CCCC(O)C(=O)N1CCC(CF)(NC(=O)CCC2CCCCC2)C1 N1(C(C)=O)c2ccccc2Sc2ccccc21.C1(=O)CC(C)(C)CC(=O)NCC(C)N1 C1(N(C(CSC)=O)CCO)CCCN(C(=O)C(C)=C2CC2)C1 c1(C(N2CCC(CNC(CNS(NC)(=O)=O)=O)C2)=O)ncnc(O)c1Cl c1(C(N(CCCNC(=O)CC2CCCO2)C(C)C)=O)noc2c1CC(F)(F)CC2 c1(NC)nc(C)ccc1C(=O)NCC(C)CNC(C1(OC)CC1)=O C1(OCC)CN(C(c2cnn(C)c2Br)=O)CC1CNC(C1CC1C(=O)N)=O.C(C)CC N1(C(C(c2ccc(F)c(Cl)c2)N)=O)CCC2OCC(=O)NC2C1 c1(OC)cccc2ccc(NC(C3CC(NCc4ccc(F)nc4)C3)=O)nc12 C1(N(C(C=CC(C)C)=O)C)CCC2CN(C(=O)Cc3cccc(F)c3)CC12 C1(C(=O)NCC2(F)CN(C(c3c(C)c[nH]n3)=O)C2)CCC12CCCO2 N1(C(CSCc2nc(C)sc2)=O)C2CCC1CN(C(C13CCCC1CCC3)=O)C2 c1(C(=O)NC(CC)CN(C(=O)C(N2CCOCC2)C)CC)cc(C)n(C)c1 N1(C(=O)COc2cc(C3CC3)on2)CCN(CC(F)(F)CO)CC1 C(=O)(C1CCSc2ccccc21)N1C(C)CN(C(=O)CCCCCC#N)CC1 N1(C(Cc2cc(C)sc2C)=O)CCC(NC(c2cc3n(n2)CCCN3)=O)C(C)C1 C1(C(=O)NC2CC(CCOC)C2)CC2CCC(C1)N2C(c1cc(C(N)=O)co1)=O N1(C(c2c(C)nc(C(C)C)o2)=O)CC(C)N(C(=O)CSCC(F)(F)F)CC1C C1(C)(NC(C(C)=C(C)C)=O)CCN(C(=O)C(C)c2ccco2)CC1 C1(NC(c2cnc(OCC)nc2)=O)CCN(Cc2ccc(OC)c(Cl)c2)CC1C N1(C(C=C(CC)CC)=O)CC(OC)CC1CNC(c1ccc(C#N)o1)=O CN1CCc2[nH]nc(C(=O)NCC3(NC(c4c(N)cc(Cl)cc4Cl)=O)CC3)c2C1 N1(S(CCC(CC)CC)(=O)=O)CCCN(C)CC1C Cc1cc(C(N2CCN(C(c3cn(C4CCC4O)nn3)=O)CC2C)=O)cc(N)c1 c1(OC)c(C(=O)NC(C)CC2CCN(C(=O)CN(C)C(=O)OC)CC2)csc1C C(=O)(C(C)(C)C(C)(F)F)NC(CCC)CCCNC(=O)Cn1cnc(C(=O)OC)c1 c1(CC(=O)NC2C(C(C)C)N(C(=O)CCC(F)F)CC2)ccc2c(c1)OCCO2 c1(C(N2C(CN(C(CC3(C=C)CC3)=O)C)COCC2)=O)cncc([N+](=O)[O-])c1 CC1(C(=O)NCc2ccc(CO)s2)CCCN1C(C1CCCC1)=O CN=C(NCC1CC1c1cnn(C)c1)NCC1(CF)CCC1 c1(CC)cc(C(=O)NCC(C)NC(=O)Cc2ccc(C)c(O)c2)cc(Cl)n1 C(=O)(C1COc2ccccc21)N1CC(C)C(NC(=O)NC2(C)CCNC(=O)C2)C1 c1(C(=O)NCCOCCNC(C(=O)N(C)C)=O)ccc(S(C)(=O)=O)[nH]1 C(C1OCCc2sccc21)N(C(C1CCCN(c2c(OC)nccc2)CC1)=O)C N1(C(c2nc(CC)oc2)=O)CC2CCC1C(NC(=O)CCC1CCC(C)O1)C2 N1(C(=O)OC(C)(C)C)CCCC1C(=O)NC12CC(CNC(=O)CCCCCO)(C1)C2 C1(CC(=O)NCC(CC)N(C(=O)CCC2CCOCC2)C)CC(C)(C)C(=O)N1 N1(C(CN2CCC(C)CC2)=O)CCC2(CC1)CC2NC(=O)CN1CCC(C)(C)C1 N1(C(C2CC23CCOCC3)C(=O)NCC(C)C)CCC(C2CC2)C1 N1(C(c2n[nH]c(C)c2N)=O)CCN(C(=O)C=Cc2cccc(CO)c2)CC1C O(N1C(=O)CNC1=O)CC(=O)OC.C1(CNC(=O)CC2(CO)CC2)CCCC1N c1(NCCOc2ccc(C)cn2)nc(NC2CC3CC(O)C2C3)c2c(ncn2C)n1 C1(NC(C2CCN(Cc3ccncc3)CC2)=O)CCC2C(CC1)C2(F)F c1(NC(CC2CC3(CN(Cc4ccn(CC)n4)C3)C2)=O)cc(C)cn2ccnc12 c1(C(N2CC(NC(C(CC)(C)O)=O)C(O)C2)=O)occ2c1CCC2 CC#CCC(C(=O)NCc1nnc(C)o1)NC(=O)C(CC)=CCCC CC(CCC(=O)N1CCCC(N(C)C(c2nn[nH]c2Cl)=O)C1)N(C)C C=C(C)CC(C(=O)N(CCCCCCNC(c1ccccc1CC#N)=O)C)OC Cc1c(C(=O)NCC2(OCC(=O)N(C)Cc3nc[nH]n3)CC2)sc2cncn12 N1(C(C(CC)n2cccn2)=O)CCC(C)C1C1(NC(=O)C(F)=CC2CC2)CC1 C(c1ccc2c(c1)OCCO2)=Cc1c(Cl)ccc(C(NOC)=O)c1 N1(C(c2cc(OC)ncc2)=O)CCN(C(c2[nH]nc(C(F)(F)F)c2C)=O)CC1C c1(C(=O)NCC2C3CN(Cc4c(OCCC)cccc4)CC32)cc(C)nc(O)n1 CCC1=C(C(=O)N2CCCC2(C)CNC(C2CC3(CCCC3)CO2)=O)CCCO1 N1(C(CCSCCC)=O)CC2CCOC2(CNC(=O)C(C)(C)CCSC)C1 c1(C(=O)NC(C(=O)NCCC(C)N(CCC)C)CO)cnn2c1OCC2.C(C)S c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)C=CC(c2ccccc2)=O)C(O)C1)=O c1(NC(C(N2C(C)CC(NC(CCOC)=O)C2)=O)=O)cccnc1F CC1CC(C(=O)Nc2ncccc2O)N(C(c2cnn(C3CCCC3)c2)=O)C1 Cc1ncc(C(=O)NC(C)CCNC(=O)CCC(=O)Nc2nccs2)n1C(F)F C12(NC(C3(CNC(C)=O)COC3)=O)CCCC1N(C(c1ccco1)=O)CC2 c1(C(=O)NCC2CCN2C(C2CN(CC(F)(F)F)C2)=O)cccc(C2CC2)c1 C#CC1C(C(N2CCC(OCC)CC2)=O)C1(C)C.c12cn(nn1)CCNC(=O)C2 C1(CCNC(C)=O)CCN(C(=NCCCCl)NCC(C2CCOCC2)C)C1 CC1CCC(NC(c2c[nH]c(=N)o2)=O)CN1C(c1cnc(O)c(F)c1)=O C(=O)(C(F)C(C)CNC(C1OCCC1(C)C)=O)N1C(C)COCC1 S(=O)(=O)(c1ccc2c(c1)CNC(=O)O2)NCc1snc(COC)n1 c1(C2C(C(=O)NCCN(C(CC3ON=C(C)C3)=O)C)C2)cc(F)cc(Br)c1 C1(CNC(c2cc(SC)oc2)=O)CC2CCC1N2C(=O)C(C)C1CCCO1 c1(C(=O)NC2(C)CN(C(C(C(CC)C)O)=O)C2)cc2n(n1)C(C)CCC2 N1(C(CC)=O)CCCCC1CNc1nccnc1C(F)(F)F c1(C(=O)NC23CC(NC(C4CCC(OC)C4)=O)(C2)C3)c(C)nn2cc[nH]c(=O)c12 n1(CC(N2CCC(Cn3cc(C(C(C)C)O)nn3)CC2)=O)cnc2sccc2c1=O C=CC1CN(C(c2cnn(C(C)C)c2)=O)CC1NC(=O)C(O)CN(C)C c1(C(N)=O)ccccc1OCC(=O)NCC=CCNC(C1CC2CC2C1)=O c1(C(=O)NC(C2CCCN(C(c3cnc(Cl)c(Cl)c3)=O)C2)C)cccc(Br)c1F CC1(C)CCCN(C(c2cnc[nH]2)=O)C1CNC(c1cc(O)cc(Br)c1)=O C1(C(N2CC(CNC(c3cc(OCC)no3)=O)C(O)C2)=O)CCCNS1(=O)=O C1(C(=O)NC(c2ncnn2C)CC)CCCN(C(c2cc(C)sc2C)=O)C1 c1(-c2nc(NC(c3cnc(N(C)C)o3)=O)sc2)ccc(C(N2CCSCC2)=O)cc1 N1(c2nnn(C)n2)CCC2(CC1)C(NC(=O)C=Cc1cnc[nH]1)CS2(=O)=O N1(C(CCNC(=O)OC(C)(C)C)=O)CC(n2cccn2)(NC(COCCF)=O)C1 c1(C(=O)NCC2C(C)(C)N(C(=O)C(O)C(F)(F)F)CC2)cc2ccccc2nn1 Cc1ccc(S(=O)(=O)N2CCN(C(=O)CN3CCCC(C)CC3)CC2)cc1C(=O)O N1(C(C(c2cnc(Cl)s2)C)=O)CCC(c2cn(CC(C)O)nn2)C1 c12nnc(N3CCN(CC(=O)OC)CC3)n1C2.C1(C(=O)OCC)CCOC1(C)C c1(NC(C2N(C(c3[nH]cc(C)c3)=O)CC(F)(F)C2)=O)cnc2cc(Cl)ccc2c1 c1(C(C)C)ccoc1C(=O)NC1(C(=O)NCc2noc(C3CC3)n2)CC1(C)C C1(NC(CC(=O)NCC#C)=O)CCC(NC(c2nc(C3CC3)n[nH]2)=O)CC1 C1(NC(=O)Nc2c(CC)cc(C(=O)OC)cc2)CCCCC1S(C)(=O)=O N1(C(c2c(OC)nccc2)=O)CCN(C(C2Cc3ccccc3S2)=O)CC(O)C1 c1(CCS(NN(C(=O)CC2CCC(=O)O2)C)=O)ccc(C(F)(F)F)cc1 N1(C(C2(S(C)(=O)=O)CC2)=O)CCC(O)CC1C(=O)Nc1cc(C#N)ccc1O C1(NC(C(C)(C)SC)=O)CCCCC1CN(C)C.C1(C(=O)N)(CF)CCOCC1 C1(C(=O)NCC2(NC(=O)C=C[N+](=O)[O-])CCCCC2)CCC2C(CC1)C2(F)F CC(C)C(CNC(=O)NCCCS(=O)(=O)N1CCCC1)CO C(CC(=O)NC(COC1CC1)CC)(C(C)OC)NC(c1noc(CC)c1C)=O N1(C(C(CC)N(C)C(c2ccc[nH]2)=O)=O)CCCC(N(C)C)CC1 C1(CCCNC(CS(C)(=O)=O)=O)CCCN1C(C1OCCC1C)=O.CNCCN C1(CCC=C)(C(=O)NC(CO)C(N)=O)CN(C(c2cnn(CC)c2)=O)C1 C1(NC(C2(C(F)F)CC(=C)C2)c2nnnn2Cc2cccs2)CCCN(C)C1=O C1(CC)(CNC(C2COC(CNC(=O)CN3CCCC3)C2)=O)CCCCC1 C(C)(CCC(=O)N1CC(C)(C(=O)N(C)Cc2ccc(F)cc2)C1)OCC N1(C(C2C(CC)N(C)CC2)=O)CC(CNC(=O)CCNC(=O)COC)CC1(C)C N1(C(C2(OCC)CCC2)=O)CC2CN(C(C3C=CCC3)=O)CC(C1)O2 C1(C(N2CCC(C(C)(C)NC(c3c(CC)nccc3)=O)C2)=O)CC2(CCO1)CC2 Cc1cc(Cl)c(NC(=O)NC(C)CN2CCC(C)CC2)c([N+](=O)[O-])c1 Cc1ccc(C(=O)NC2CC(CNC(C3(C4CC4)CCC3)=O)C2)n1C C1(OC)CN(C)C(C)(C(N2CC(CNC(=O)C(c3cccc(Cl)c3)O)C2)=O)C1 N1(C(C2C(C(=O)NCCC#C)C2)=O)CCC(C)(CN)C1 c1(C(=O)NCCOC2CCN(C(C(C)n3ccnc3)=O)C2)cnn2c1OCCC2 C(=O)(CS(=O)(=O)C(C)C)N(CC(C)N(C(c1ncnc(C)c1C)=O)C)C N1(S(c2c(C)n[nH]c2C)(=O)=O)CCN(c2ccccc2)CC2(CC2)C1 C(C(C)(C)CCl)(c1nnnn1CC(F)F)NC(CCCOC)C C1(NC(c2cccnc2)=O)CN(C(=O)CC2CCCC(F)(F)C2)CC12CC2 N1(C(Cc2cccc(C)c2)=O)CCC2(CC2C(N2CC3COCC3C2)=O)C1 N1(C(C2(C(CC)=O)CC2)=O)CC(COC)(NC(C2(F)CCOC2)=O)C1 C1(n2cc(CC(C=C)O)nn2)CC2CCC1(NC(=O)COC(C)CC)C2 CCC(CN=c1[nH]nc(Cl)cc1N(C)C)N1CCOCC1 C(c1cncn1C)=CC(N1CCCC(N(C)C(C2(CC(F)F)CCC2)=O)C1)=O C1(C(=O)NCCCc2ncco2)CCC(C2CC2)N1C(C1CCC(CO)CC1)=O N1(CC(=O)NCC2(OC)CN(C(c3ccc(N)cc3C)=O)C2)CCS(=O)(=O)CC1 c1(C(F)(F)F)ccc(-c2cncc(CN3CCOCC3)n2)cc1 c1(C(N(CCOCCC(=O)NC(C)CCO)C)=O)ccn2ccnc2c1 c1(C(=O)NCCN(CCC)C(C2(N(C)C)CCCSC2)=O)cnccc1Cl C1(C(C)(C)C)C(NC(=O)C(=O)NC2CC2)CCN1C(=O)CC1(C(F)(F)F)CC1 C(C1=CCCN(C)C1)NC(CC1(C)N(C(C2CCC(C)O2)=O)CC1)=O N1(C(C(C)C(F)(F)F)=O)CCCCC12CN(C(c1cn3c(n1)SCC3)=O)C2 c1(C(N2CC(OC)C(NC(=O)C(C#N)C3CC3)C2)=O)cc2cnccc2cc1F C(=O)(CCCC(=O)NCC1CCN1CC(=O)Nc1ccc(C)cc1C)NC Cc1ccc(C(C)(C)CC(=O)NCCOCCN(C(=O)C(C)C2CCC2)C)cc1 C=C(C)C(CC(=O)NC1CCC(F)(CNC(c2cc(O)n(CC)n2)=O)C1)OCC C1(C2(NC(=O)Cn3nccn3)CC2)CCCN1C(=O)Cc1nccs1 N1(C(c2cc(C)cc(C)c2)=O)CC2(CCCC(CNC(C3CS(=O)(=O)C3)=O)O2)C1 CC1(C)CC(=O)NCC1C(=O)NCC1CN(C(c2sccc2F)=O)CC1(F)F N1(C(=O)Cn2ccccc2=O)CC(C2CN(C(C3C=CCCC3)=O)C2)C1 c1(C(N(C(CNC(=O)COCP(C)(C)=O)C2CC2)C)=O)c(F)cc(F)cc1Cl C(C(CC)CC(C)C)NC(C1(CO)CCN(C(c2c(C)con2)=O)C1)=O C(=O)(C1COc2ccccc21)OCC(OC)(NC(c1ccn(C)c1)=O)OC c1(C)cnc2sccn12.N1(C(C2C(CN)C2(C)C)=O)CCCC(C(=O)OCC)C1 c1(C(=O)NC(CCSC)C)oc(CNC(C2CNC(=O)C2)=O)cc1C Cc1ccc(=O)n(CC(=O)N(CCCNC(C2CC2[N+](=O)[O-])=O)CCO)n1 c1(CC)ccoc1C(=O)NCC(CC)NC(=O)C(=O)Cc1cccs1 C1(NC(C2CCCO2)=O)CCC2CN(Cc3ccc(Cl)c(F)c3)CC2C1 c1(C(N(CCNC(CC2N(CC)CCOC2)=O)C)=O)cccc2c1OC(C)C2 c1(CCN(C)CCn2cc(CC(=O)O)nn2)cscc1Br C12(NC(c3cnns3)=O)CCC(CC1)N(C(=O)C=Cc1ccccc1F)C2 c1(CNC(C2C(C(=O)NC3(CC)CCOCC3)C2)=O)ncc(Br)cc1C c1(NCc2cc(OCCOC)c(Br)cc2)cc2c(o1)CCCNC2=O CCC(O)C(C)C(=O)NCC1CC(NC(c2cnnn2C2CC2)=O)C1 c1(SCC(=O)NC2CCC(C(=O)NCCNC(C)=O)C2)ccc(O)cc1 Cc1ncc(Cl)cc1C(=O)NC1CN(C(=O)CC2CSC2)C2CC12 C1(C(N(C2CCN(C(=O)C(O)P(C)(C)=O)CC2)CC)=O)CCC(=O)N(C2CC2)C1 c1(OC(F)F)nccc(=NC2CC(NC3CCN(C4CCCC4)C3)C2)[nH]1 C(=O)(C(C)(C)C(=O)NCC1CCN(C(=O)Cc2cncc(C)c2)C1)NC C(=O)(CC(C(F)F)C(C)(C)C)N1CCCC(CCNC(c2c(C)cco2)=O)C1 C1(C(N(CC(=O)OC)CC=C)=O)CC(CCNC(=O)C(C)c2cc[nH]n2)C1 C1(C(=O)NC2(C(C)C)CCC2)(NC(=O)C=C2CCC2)CCCC1C Cc1cc(C(=O)NCC(CO)NC(c2nccn2C)=O)c2cccc(C)c2n1 c1(CC(=O)NC2C(NC(c3ccn(CC)n3)=O)COC2)c(F)cncc1Cl CC1CN(C(=O)Nc2nc(N3CCCC3)ncc2Cl)CC(C)(C)O1 CCC(O)C(C)(C)C(=O)NCC(c1ccc(F)cc1F)NC(c1ccc(C)s1)=O C1(NC(c2ccc(C#C)nc2)=O)CCSC12CN(C(=O)C(C)C)C2 Cc1cccc(N2C3C(CCC3)CC2=O)c1.C(=O)(COC(=O)CO)NCC(C)C N1(C(CCNC(C)=O)=O)CC(C(=O)Nc2nc(Br)ccc2Cl)CC(F)C1 C1(OCC(C)C)CCN(C(C2CCOC2CNC(c2c[nH]cc2C)=O)=O)C1 c1(C(=O)NCCC(=C)CNC(=O)C(C(C)C)OCC)cc2c(cc1N)CCC2 N1(CC)C(=O)CC(NC(=O)N(C)C2CC2)C1c1ccccc1OC C(=O)(CCC(C)(C)C#N)NC1C(C)CN(C(C2CCN(CC(F)F)CC2)=O)C1 N1(C(C(CC#C)(C)C)=O)CC2CC(NC(=O)CN3CCCC3CO)C(C2)C1 C1(C)(C(=O)NCCOCCN(C)C)C=CCN1C(c1ccnc(CO)c1)=O C(CC(=O)OC(C)(C)C)(C(C)C)N(CC(C1CCCOC1)O)C(=O)OC N1(C(c2cccc(CNC(CC=CC=C)=O)c2)=O)CCCCC1C=C C(=O)(CCC(C)(C)C#N)NCCC1C(C)CCCN1C(=O)Cn1ccnn1 O(NC(=O)C(Cc1ccc(F)cc1)N1CCC(COCC)C1)CCC#C.C(C)(C)(C)O c1(CN2CCC(NC(C3CC34CCOC4)=O)(CF)C2)cc(Br)ccc1Cl N1(C(C(CC)(CNC(C2Cc3nccn3C2)=O)CC)=O)Cc2nncn2C(C)C1 Cc1cnc(C(=O)NCC2CC(C)N(C(=O)C(C)(C)n3cccn3)C2)nc1 c1(OC)cc(CN2CCOCC2CC(=O)Nc2ccccc2C#N)ccc1C C1(NC(CCCC)=O)CCN(C(=O)CN(C)C(=O)C2CC2)CC1C(N)=O c1(C(=O)NC(CCCC)C(=O)N2CC(OC)CC2CF)ccn2ccccc12 C1(CC(N2C(C(C)C)CCCC2)=O)CCN(C(c2ccc(F)cc2F)=O)C1(C)C C1(C#C)(C(=O)NCCC(C)N(CCC)C)CCN(C(=O)C(C(C)C)C(C)C)CC1 N1(CCCC)CCN(CC#N)C(CS(C)(=O)=O)C1.c1(C=O)c[nH]nc1CC(C)(C)C C12(CN)CCCC1C2(F)F.n1(CC=C)cc(C(c2nnnn2CC(F)F)(C)N)nn1 C1(CNC(CC2CCCC(OC)C2)=O)COCCN(C(c2ccccc2)=O)C1 C1(C(N(C)Cc2ncnn2C)=O)CN(C(C2CCCO2)=O)CCC1(C)C c1(C(N2C(C(=O)NCC3(CC)CCCO3)CC2)=O)cc(N)cc(F)c1 N1(C(C2(C)CCCO2)=O)Cc2n[nH]cc2C1C(=O)N1Cc2ccncc2C1 N1(C(C(C)(C)OC)=O)CC(NC(c2csc(=NC)[nH]2)=O)C(n2cccn2)C1 C1(CC(=O)NCCC(=O)N(C)CC2(CN3CCCC3)CC2)CCS(=O)(=O)CC1 C12(C(=O)NCCC3CCN(C(=O)COCC4CCCO4)CC3)CCCC1C2(F)F CC1(CNC(=O)C(CO)NC(=O)CCC2CC2)CC2CC2C1 N1(Cc2ccc(OC)cc2F)CCC2C1CCCN2c1ccnc(NC(C)=O)n1 C1(CCNC(C2(CC=C)CC2)=O)CSCCN1C(c1cnn(C)c1)=O c1(C(=O)NCCN(c2nccc(C(F)F)n2)CCOC)nc(OC)ccc1OC C1(C(N2CC(C3CCN(C(CCOCC#C)=O)C3)OCC2)=O)CC2(CCO1)CC2 c1(C(=O)NCCN(C(CCCCOC)=O)C)cn(C(C)C)c(=O)nc1O c1(C(=O)NC2C(C)N(C(c3ccccc3F)=O)CC2)[nH]c2ccccc2c1Br c1(C(=O)OCC(C)SCC(c2ccc(C(C)C)cc2)=O)ccc(F)cc1Cl Cc1ccccc1C(=O)NCC1CCN(C(c2ccc(NS(C)(=O)=O)cc2)=O)C1 C1(C(N2CCCCC(CNC(c3ccc(O)nc3)=O)C2)=O)CC2(CCCC2)CO1 C1(C(=O)NCc2nc(N(CCOCCOC)C)sc2)CC(c2ccccc2)=NO1 C1(CC)(NC(=O)CC(C)(C)O)CCCN(C(=O)C(C)(C)CC(=O)OC(C)(C)C)C1 Cc1cc(-c2cn(C(C)C(=O)NC3CCOCC3C)nn2)cnc1C CCC(C)(C)CC(=O)N1CC(O)(C(C)OC)C1.c12csc(n1)C(C)NC2=O C1(C(=O)NCC2CCN2C(=O)CC2CC2(Cl)Cl)CC12CCc1ccccc12 c1(C(=O)NCC2CC2NC(c2cnns2)=O)cccc(CCO)c1 C(CC(=O)N1CCC(C)(NC(N)=O)C1)(C(F)(F)F)N(C(CCCC1C(C)C1)=O)CC c1(CC)ccccc1C(CNC(c1c[nH]nc1C)=O)NC(c1ccccc1)=O C1(CNC(CCC(CC)CC)=O)CN(C(C2C=CC=CC=C2)=O)CC2(CCC2)O1 C1(CN2CCCC(C(C(=O)OC)CNC(=O)OC(C)(C)C)C2)CCC2(CC1)CC2 c1(SCC(C)C(=O)NCCNC(c2cocn2)=O)ccc(Cl)cc1 CCCC(O)C(CO)NC(C1CCC(C)N(C(=O)CNC=O)C1)=O N1(C(c2ccn(CC)n2)=O)CC(CNC(C2CCC(C)O2)=O)CC12CCOCC2 c1(OC)ncc(C)c(C(=O)NC(C)C(c2ccccc2)NC(=O)CC#N)c1Cl C1(C(N2CC(C(F)(F)F)(NC(C=C(C)C)=O)C2)=O)CC(=O)CC(=O)C1 Cc1cccc(C(F)(F)C(=O)N(C)CC2CN(C(C3CCCC34CC4)=O)C2)c1 C1(NC(CC2(C)CCC2)=O)CC(C(=O)NC2CC3CCC2CC3)C12CCC2 N1(C(C(C)(C)O)=O)CCC2(CCCN(C(=O)C3Cc4c(Cl)cccc43)C2)C1 c1(OC)ncnc(C(N2CCCCC2CN(C(=O)Cn2nnc(=N)[nH]2)C)=O)c1F c1(CC)oc(C)cc1C(N1CC(NC(C2CCC(F)C2)=O)C(F)C1)=O c1(C(N2C(CCC)CN(C(=O)C=Cc3cc[nH]n3)CC2)=O)nc(O)nc(O)c1N C(=O)(C(C)C(C)(F)F)NCC(CN(C(Cc1c(C)nc(C)s1)=O)C)(C)C CC1CCN(C(c2ccc3ncccn23)=O)CCN1C(C1CNC(=O)C1)=O C1(C(=O)NCCSCCCO)C=CCCN1C(c1ccc[nH]1)=O C1(C(N(C)Cc2ccn(CC)n2)=O)CCOCCN1C(=O)CCn1ccnc1C c1(OC)ccc2c(c1)OCCC2N(C)C(=O)NCc1ccc(C)c(OC)c1 C(=O)(C#CC1(C)CCCO1)N1CC(CNC(c2ccc(OC)nc2C)=O)C1 c1(C(N2CCCC2(C)CNC(C2=C(C)OCC2)=O)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] CCC(CC(=O)N(C)CC1(NC(=O)CC2CC(CC(C)(C)C)C2)CC1)C(C)C CC1CCN(C(C2(NC(=O)CCc3cncnc3)CCC2)=O)CCC1(F)F c1(C(=O)NC(C(=O)NCCc2cn(CC)nc2)C2CCCO2)ccc(O)cc1 C(=O)(C1CCCc2nn[nH]c21)NC(C(C)C)(C)CNC(=O)Cc1nn(C)cc1Cl CCCCC(C(=O)OCC1CCC=CCC1)ON=C(C)C c1(OC)ccc([N+](=O)[O-])c(C(N2CC(NC(=O)CCCN(C)C)C(C#N)C2)=O)n1 C(=O)(CC(C)N(C(c1ccccc1)C(=O)Nc1c[nH]c(C)c1)C)OC C12(NC(C(C)NC(N)=O)=O)CCC(CN(C(=O)COc3ccccc3O)C1)C2 C(=O)(C(C(C(C)C)OC(=O)C(C)N(CC)CC)N(C1CCCOC1)C)NC(CC)C CC(C)C(O)C(C)C(=O)N1CCC(C)(CNC(c2ccc(S(N)(=O)=O)s2)=O)CC1 c1(C(N2CCC(Cc3onc(C(C)C)n3)C(F)(F)C2)=O)ccc2n[nH]cc2c1 C1(C(=O)NCCCN(C(C(CC)CC)=O)CC2CCCC2)CCCCC1N=[N+]=[N-] CP(C)(=O)c1cnc(C(N2CCCC(CNC(c3ccc[nH]3)=O)C2)=O)nc1 C1(NCc2cccc(C(N(CCC#C)CCOC)=O)n2)OCCOC1(C)C C1(CCCC(N2CCC(NC(CCn3ncc(C)c3)=O)C2)=O)CCCC(=O)N1 c1(C(N2CC(NC(c3c(CC)c[nH]c3)=O)C(OC)C2)=O)ccc(C)c(F)c1F N1(C(c2cccc(OC)c2O)=O)CCN(C(C2CC2C(F)F)=O)CCC1C C12(NC(c3cc(C(C)(C)C)no3)=O)CCC(NC(C3(C)CC=CCC3)=O)(CC1)C2 N1(C(c2ccc(CCOC(C)(C)C)cc2)=O)CC2CCCC2(C(F)(F)F)C1 c1(C(=O)NC(CC(C)NC(c2c(C)noc2)=O)C)cc(F)c(Br)cc1N c1(NC(C2CC2NCc2c[nH]c3ccc(Br)cc23)=O)c(Cl)cc(Cl)cc1[N+](=O)[O-] c1(N2C(CNC(c3ccc(SCC)cc3)=O)CCC2)nc2cccc(C)c2o1 C1(NC(=O)CCCC2(NC(=O)CSC3CC3)CC2)CCOCC1F Cc1cnc2nc(C(=O)NC(CNC(c3n[nH]c(C(C)(C)C)n3)=O)CO)nn2c1 c1(NC(C(C(C)C)C)CNC(=O)C(n2cc(Cl)cn2)C)ccnc2ncnn12 c1(CC)cc2ccccc2cc1S(=O)(=O)N1CCSCC1c1nccs1 C(C(C)(C(=O)NCC1(F)CC(NC(=O)C=CC2CC2)C1)OC)OC c1(C(=O)NCCC(C)NC(=O)Cn2cnc(=N)[nH]2)ccc(C(F)F)c(F)c1 C1(NC(C2CNC(=O)N2)=O)CN(C(c2nccc(Cl)c2F)=O)CCC12CCC2 c1(C(=O)NCC2(C(C)NC(=O)Cc3nonc3C)CC2)cn2ccsc2n1 C(=O)(C(CNC(=O)CC1(N(C)C)CCC1)CCC)NC(CC#C)CC CN1CCC(N(C)C(c2conc2C(C)NC(=O)CCN(C)C)=O)C1 C=CC1(C(=O)NCC23CCC(C2)N(C(C2CC(C(C)C)C2)=O)C3)CCOCC1 c1(CCC)ccc(C(N2CCC(CN(C)C(C3CCCO3)=O)CC2)=O)cc1 C(CCSC)(C(=O)N1CCC2CC12)NC(C(C1CCCC1)OC)=O C(C(CC(C)C)NC(CC)=O)N(C(=O)OC(C)(C)C)CCC.C1(=O)C=C(C)CN1 C1(NC(c2ccc(COC)o2)=O)CCN(C(=O)CCC(C)C)CC1CO c1(OCCCC(=O)NC(C2CCN(C(=O)CN(C)C)CC2)C)ccc(F)cc1 c1(C(=O)NCC2CC(NC(CN(C)C)=O)C2)ccc2nccn2n1 C1(CNC(C=CC(=O)N(C)C)=O)CCCCN(C(c2cc[nH]n2)=O)C1 CC1(C)C(=O)Nc2ccc(S(=O)(=O)NC3CC3C(=O)NNc3ccc(F)cc3)cc21 c1(CNC(CCNC(C(C)(C)c2cnn[nH]2)=O)=O)ccc(O)c(F)c1 Cc1nc(C=CC(=O)NC2CCN(C(C3CC(=O)N(C)C3)=O)C23CC3)[nH]c1C C(=O)(C(C)C(C)NC(=O)NCC1(OCCO)CCOCC1)OCC C1(C(=O)NCCN(C(=O)Cc2cccc(C(F)(F)F)c2Cl)C)CCCC(C#N)C1 C1(CNC(c2c(C)cno2)=O)CN(C(c2cnc(S(C)(=O)=O)s2)=O)CCC1(C)C S1(=O)(=O)c2ccccc2CN1.c1(C(OCOCC)=O)ccc(F)cc1F c1(CC(=O)NCC2C(NC(=O)CN3CCOCC3)CC2O)csc(Cl)n1 N1(C(C=C(CC)C)=O)CC(NC(=O)COc2cc(Cl)ccc2C)CC2(CC2)C1 C(=O)(C(F)(F)CCCC)N1CCC(N(CC#C)C(C2CCCCCN2C)=O)C1 Cc1nc(NC(C)(C)CCNC(c2cccc([N+](=O)[O-])c2)=O)c2cnn(C)c2n1 c1(C(=O)NCCCC2N(c3nnc(C)s3)CCC2)ccc2ncsc2c1 N1(C(C(C)(C)NC(C)=O)=O)CC(CNC(c2cccc(C)c2)=O)C2(CC2)C1 [N-]=[N+]=NC1CN(C(=O)CC2CCN(C(c3cnc(S)nc3)=O)CC2)CC1O C(CN=c1[nH]c(N(CC(=O)N(C)C)C)nc2c1CSC2)(C(C)C)OC C1(NC(C2(CC)CC2)=O)CCC(CNC(=O)CN(C)C(N)=O)C1.c1ccccc1 c1(CN2CC(C)(C(=O)Nc3c(OC)cccc3)OCC2)cn2c(n1)COCC2 C1(C(=O)NCCCN(C(=O)CCCNC(=O)OC)CC)CCNC(=O)C1 CCCC(C)CC(=O)NCC1CC(OC)CN1C(c1ccc(COC)cc1)=O c1(C(N(CC(C)NC(C(CC)O)=O)C)=O)ccn(CC(F)F)c(=O)c1 C1(N(CC(=O)NCC23CC(NC(CCCOC(C)=O)=O)(C2)C3)C)CCS(=O)(=O)C1 Cn1cc(NC(=O)C(N2CCC(Oc3cccc(Cl)c3)CC2)=O)c(Br)n1 c1(OCC=C)cccnc1C(=O)NC(CNC(=O)C(Cl)=CCl)C(C)C N1(C(=O)NC(CCc2ccc(OCC)cc2)C)CC(=O)Nc2ccncc21 N1(C(C(=O)N(CCN(C(C=CCOCCCOC)=O)C)C)C)CCNC1=O c1(CCC(=O)NC(C(C)C)CNC(C2CC(C#N)C2)=O)ccc(F)c(F)c1 C1(NC(C2CCCN2CC(F)(F)F)=O)(CO)CCCN(C(C2C3CCCC23)=O)C1 C(=O)(C(F)(F)C(C)c1ccccc1)NCCC(C)NC(C=C(C)C)=O c1(CC(N2CC=CC(NC(C(CC)COC)=O)C2)=O)cc(Cl)ccc1O C1(N(C(=O)CC(C)F)CCC)CCN(C(c2csnc2C)=O)CC1 CCC(C(=O)N1CC(C(n2cc(Br)cn2)c2nn[nH]n2)C1)c1cccnc1 c1(C(N2CCC(CN(C(=O)CC34COC(C)(C3)C4)C)C2)=O)cc2cccnn2n1 C1(OCC)CN(C(=O)CCCC2CCCC2)CCS1.C12(O)CN(C1)C2=O C1(CNC(COCCN(C)C)=O)CCCN1C(=O)CCn1cncn1 N1(C(C2N(C(Cc3c(C)nn(C)c3)=O)CCC2C)=O)CCCC2(CC1)CC2 c1(N2CC(C)C(CNC(=O)Cn3cc(Cl)cn3)CC2)ncnc2cc(C3CC3)nn12 CC1CC(NC(c2csc(-c3ccsc3)n2)=O)CN(C(=O)C=CCO)C1 N(C(=NCc1occc1C)N1CCC(C)C(F)(F)C1)CCC(C)=O c1(CC)nc(C)c(C(=O)NCCCC2(NC(=O)CSc3nc[nH]n3)CC2)s1 Cc1cnc(NCc2cnsc2)c(S(=O)(=O)NCC(c2cccs2)O)c1 c1(C(=O)NC2(C)CCN(C(c3[nH]ncc3C#N)=O)CC2)cc2cccc(O)c2[nH]1 c1(C(N2CCC3(NC(c4c(CC)ocn4)=O)C(C2)C3)=O)cn2cc[nH]c(=O)c2n1 Cc1cnc(C(=O)N(C2CN(C(c3ccn(CCF)n3)=O)CCC2O)C)cc1C c1(C(=O)NC(CN(C(c2c(OCC)ccs2)=O)C)C)ccc(Cl)c(F)c1 CCCC(C)(CCC)C(=O)N1CC2CCC1CN2C(=O)C(c1ccccc1)F CC(C)(C)C(C#N)C(=O)NCC1CCCC(CNC(C2CN3CCN2CC3)=O)C1 c1(NC(=O)Nc2c(C(=O)OCC)c(-c3ccccc3)no2)nccc(Cl)c1F C1(N(C(COCC(C)C)=O)C)CN(C(c2nn(C)c(Cl)c2Cl)=O)CCC1C c1(CC)ccccc1OCC(N1CCC(NC(=O)Cc2ccnc(O)c2)C1)=O c1(C(N(C2CCC(NC(COC)=O)C2)C)=O)nccc2[nH]ccc12 C1(C(OC)OC)CCCCN(C(=O)NCCn2cncc2-c2ccccc2)C1 C1(C(=O)NCCCCCNC(c2c(C)ncs2)=O)COCC2(CCC2)O1 c1(C(N2CCC(N(C(c3cc(Br)c[nH]3)=O)CC)C2)=O)ccc2oc(=O)oc2c1 N1(C(C(C=C)(C)C)=O)CC(C2CCCN(C(c3cc4c(C)n[nH]c4cn3)=O)C2)C1 c1(C(=O)NCC2CCCN(C)C2)ccc(-c2cccc(C(F)(F)F)c2)c(F)c1 C#CCC(C)(C(=O)NCc1nc(N(C)C)no1)NC(C1COC(C)C1)=O C1(CNC(CCC#C)=O)CC(C(F)(F)F)CCN1C(c1cncc(C2CC2)c1)=O N1(C(CNC(=O)CCCCO)=O)CCC2(C1)CN(C(C1CC1Cc1ccccc1)=O)C2 C1(NC(c2nnn(C(C)(C)C)n2)=O)CN(C(C2CCCCS2(=O)=O)=O)CCC1F CCC(CC(C)C)C(=O)NCC1CC(O)CN1C(=O)Cc1cnc(C)s1 N1(C(C(COC)N(C)C)=O)CCC2(C1)CN(C(C1CC1C(=O)OCCO)=O)C2 C1(C(=O)NC2(C(N(CC(C(C)C)C)C)=O)CCOCC2)C2CCC(F)(F)C12 C1(C(N2CC(Nc3cc(O)ncn3)CC(C)C2)=O)CNC(=O)C(C)(C)C1 C12(CNC(COC(CC)C)=O)CCCC1N(C(=O)Cc1ccc(F)cc1)CC2 c12cc(nn1CCO)C(=O)N2.c1(C(N2CCC(OCC)C2)=O)sc(CC)nc1C N1(C(C(C)OC(c2cc(OCC)ncc2)=O)=O)CC2CCCC2(OCC)C1 Cc1c(C(=O)NC(C)CNC(c2cnc(C(C)(C)C)s2)=O)sc2cccc(F)c12 CC1(C)CN(C(c2cccc(C(N)=O)n2)=O)CC1NC(C1CN2CCN1CC2)=O c1(C(=O)Nc2n(CCCC)ncc2)ccc(-c2cncc(-c3cccs3)c2)cc1 C1(O)(C(C)NC(C2C(C(C)O)C2)=O)CCN(C(C2CCN(C)C(=O)C2)=O)CC1 CCCCCC(C)(CC)C(=O)NC1CC2CCC(C1)N2C(C1CC1CCOC)=O CC(C)C(C(C)NC(=O)CCCc1csc(=N)[nH]1)NC(c1nc(Cl)cs1)=O c1(C(N2CCC(C)(CNC(C3(C)CS(=O)(=O)C3)=O)C2)=O)cc2ccccc2s1 C1(OC)CC(CNC(=O)Cn2cc(Br)cn2)N(C(=O)CC2CC2(Cl)Cl)C1 C1(NC(CCC(C)SC)=O)CCN(C(=O)CCC(C)(F)F)CC1OC C1(C(=O)NCc2scc(C)c2)CCN(C2CN(S(C)(=O)=O)C2)CC1 C1(C(N(C(CC#C)C)C)=O)CN(C(C2(C)SCCCS2)=O)CC1F C(=O)(CCCCC(=O)N1CCC(C)(C(=O)NCC2(CO)CCCO2)CC1)OC c1(C(=O)NC(CN(C(c2ccn(C(CC)CC)n2)=O)C)C)csc2nccn12 C1(CCC)CN(C(=O)CC(=O)OC)CCN1C(=O)C(c1ccc(C)o1)C Cc1noc(N)c1C(N1CC2CC2(C(=O)Nc2csnc2C(C)C)C1)=O C12(CC)CN(C(=O)COc3ccc(Br)cn3)C(CNC(=O)CCF)(C1)C2 C(C(C)C(=O)N1CC(C(=O)NC(C)CN2CCCC2)(OC)C1)OC.CCOCCO C(CN=c1[nH]c(N2CCCC(OC3CC3)C2)nc(=N)[nH]1)c1n(C)c(Cl)cn1 N1(C(C(C=C)CC)=O)CC(C)(CNC(=O)C(C(C)C)C(C)C)CC1(C)C CC(C)(CNC(=O)CCOc1ccccc1F)CCNC(c1ccc(F)cc1)=O C(CC(C(=O)NC(c1ccncn1)C)NC(c1ccn(C)c1C)=O)OC c1(C(=O)NCCC2CCCN2C(=O)CCc2cc[nH]n2)cc(C2CC2)nnc1O n12cc(nn1)CC2.C(CCNC(=O)COCCCF)N(C(N)=O)CCO c1(C(=O)NCC#CCNC(Cc2ccc(OCC)nc2)=O)c(N)cc(F)cc1F C1(C(=O)Nc2ccc(CS(=O)(=O)NC)cc2)CCC2(CC1)CC2N C1(N(C(=O)Cc2cccc(NC(C)=O)c2)CC)CCN(C(=O)C=C(C)C)CC1C C1(C(=O)NC(C)(C)CC=CC(=O)NCC(C)(O)C2CCCC2)Cc2nccn2C1 C12(CNC(c3nc(C)sc3)=O)CCC1CN(C(=O)COc1ccc(F)cc1)C2 Cc1cc(C)c(C(=O)N(CCC(C)NC(=O)CC2CCC(=O)N2)C)[nH]1 CC1CCOCCN1C(c1cc(CNC(c2c[nH][nH]c2=N)=O)nn1C)=O N1(CC(CC)OC(=O)C(C)C(O)C(C)C)CCc2ccccc21.C1(=O)C(C)N1 N1(CCC2(CNC(Cc3cn(C)nc3)=O)CC2)CCN2C(=O)NCC2C1 c1(C(=O)NC23CC(CNC(C4CCC(=O)C4)=O)(C2)C3)cnn2ncccc12 c1(C(=O)NCC2CCCN(C(C3C(C#C)C3)=O)C2)cc(Br)ccc1N N1(C(CCN(C(C)=O)C)=O)CC2CCC1C2NC(=O)CN(C)S(=O)(=O)N(C)C CC(CCC(C)(C)C)C(=O)N1CCC2(C1)CN(C(C1CC(O)CN1C)=O)C2 c1(C(=O)OCCCc2ncc(Br)cn2)ccccc1-c1nc[nH]n1 C1(C(N2C(CC(=O)Nc3cccc(CC)c3)CCC2)=O)CC2C(C1)C2(F)F Cc1ccc(S(=O)(=O)N2CCCOC(CNC(=O)C(O)c3ccsc3)C2)cc1 CC1CC(NC(c2ncnc(O)c2Cl)=O)CCN1C(=O)CCCc1ccccc1 C#Cc1cnc(N2CCC(CNC(c3csc(O)n3)=O)C2(C)C)nc1 C(C(=O)NCCCN(C(c1cc(C(C)(C)C)n(C)n1)=O)C1CC1)(C(C)C)SC Cc1nccnc1C(=O)NC(C1(O)CN(C(c2cncnc2C2CC2)=O)C1)C N1(C(c2c(SC)cccc2)=O)CC2CN(C(=O)CC3CCCC3O)CC2(C)C1 N1(C(Cc2noc(C)c2C#N)=O)CCN(C(=O)C(C)(C)C(F)F)C2(CCC2)C1 c1(Cn2cc(CC(C)O)nn2)cccc(CC2N(C(C(CC)O)=O)CCC2)c1 c1(C(=O)NC2CCN(C(CC3OCC(C)(C)C3)=O)C2)coc2c1CCCC2 c1(N2C(C(C)(C)C)CCC2)nnc(SC2CCS2(=O)=O)n1CCC#N C1(CC(C(=O)OCC)O)CCCN(CCCCCC#N)C1 c1(N2CC3C(CNC(=O)CSC(F)F)C3C2)nc(Cl)nc2c1S(=O)(=O)CC2 O=C(CCCc1nccs1)NCC1CCC(NC(=O)Cc2ccns2)C1 Cc1cc(C(=O)NC2(C(=O)NCCC3CCCO3)CC2(C)C)nc(O)c1 c1(C(C)NCC2CCC(F)C2)ccc2c(c1)CCC(C)(C)O2 C#Cc1ccc(C(N2CCC(C)(CNC(=O)C(C)=C(C)C)C2)=O)cc1F C1(C(=O)NCCCSC)(CC)CCCN(C(=O)CNC(C)=O)C1 N1(C(CC2CC(OC)C2)=O)CCN(C(=O)C(=Cc2cncn2C)F)C(CO)C1 C(N=c1[nH]nc(C2CC2)s1)C1(CN(C(C2CCCC23CC3)=O)C2CC2)CCC1 c1(OC)cccc(CN2CCN(C(=O)C(C)(C)C(=O)O)C(CO)C2)c1OC Cc1cc2[nH]c(=NC(C)CCN3CCN(C)CC3)sc2cc1C#N.C1CCNC1 c1(C(N2CC(CNC(C3=C(C)OCC3)=O)OCC2)=O)cccc2c(Br)ccnc12 c1(C(N(C)CC2CCN(C(CCCNC(C)=O)=O)C2)=O)ccc2c(c1)COCO2 C(=O)(C1COc2ccccc21)NCC1(NC(CC2C(C)C2(F)F)=O)CCC1 N1(C(c2cc(C(N)=O)oc2)=O)CC2(CCN(C(c3cccc4nonc34)=O)C2)C1 C1(NC(=O)CC(F)F)CC(NC(c2cnnc(O)c2)=O)C(O)C1 c1(CC(N2CC(NC(C(c3ccc(O)cc3)(C)C)=O)C2)=O)cc(O)nnc1O Cc1c(C(N2CC(NC(C3CC(C)(C)C3C(F)(F)F)=O)C2)=O)sc2ncnc(N)c12 C1(OC)CC(F)CN(C(C2CC(=O)CN2C(C2(F)CCOCC2)=O)=O)C1 N1(C(CCC2(C#N)CC2)=O)CCCC(c2cn(-c3ccccc3)nn2)C1 c1(C(N(C2C3CN(C(CC(CC)SC)=O)CC32)C)=O)cc2cccnc2o1 C(=O)(CCCCCCn1cc(COC2CCOC2)nn1)NCCC(CCC)C C(C)(CC(=O)N1CCC2(CCN2)CC1)(C(=O)O)N(C)C CC(O)C(C(=O)NCC12CC(CCO1)C2)NC(c1cnc(S)nc1)=O N1(C(c2ccc(CC)cn2)=O)CCC(NC(c2c[nH]nc2OC)=O)C(CO)C1 c1(C(C)C)cc(C(=O)N(CCC(C)(C)NC(C2(N3CCOC3=O)CC2)=O)C)no1 CON(CCC(=O)NC(C)CCO)C(=O)C12CCC(C)(C1)OC2 N1(CCC)CCCC(C2CCCN(CC3(CC(=O)OC)CCCC3)C2)C1 C1(CC(N2CC(NC(CSS(C)(=O)=O)=O)C(O)C2)=O)CCCC(C)(C)C1 C1(N(C(C=NOC)=O)C)CCN(C(=O)C=Cc2ccsc2C(F)(F)F)CC1C C(C(C)C(=O)N(CCCNC(C1CCCC1O)=O)C1CC1)SC C=CCC(CC)C(=O)NC(C1CN(C(=O)CCc2nc(-c3ccco3)no2)C1)C c1(C(N2CCC(OC)(CNC(C3CCCN3C)=O)C2)=O)cc2ccccc2o1 CCC(O)C(C)C(=O)NCC1CCCCN1C(C1CCCN1C1CC1)=O C1(F)(CNC(C2CCC(C)(C)C2)=O)CCCN(C(C2(C)CC2(C)C)=O)CC1 O(C1CCC(=O)c2ccccc21)C(=O)CCC1CCOC1.c12ccc(cc1)oc2=O C1(NC(CCCc2ccc(OC)cc2)=O)C2CC1CN(C(c1nn[nH]c1Cl)=O)C2 c1(C(=O)NC(C#C)C)oc(CNC(C2CCC2C#N)=O)cc1C C(CC(C)C)(C(=O)NC12CCC(CC1NC(C1C3CC4C(C3=O)C14)=O)C2)OC O=C(CC(F)(F)c1ccccc1C(F)(F)F)NCCCN1CCCC1C(F)(F)F C1(N(C(=O)CC2CCNC2=O)C)CCCN(C(=O)Cc2cccc(O)c2)CC1 c1(CN(C(C(=O)OCC)=O)C(C)COC(c2ccccn2)=O)ccccc1F.C(C)(C)(C)O c1(NC(C(CC)N(C(=O)C(C2CCCCC2)O)C)=O)ccc(C)nc1 N1(C(c2c(F)ccc(OC)c2)=O)CC2(C1)SCCC2NC(=O)CC(C)C1CC1 c1(C(=O)NCCN(CC(C)O)C(c2cnn(C)n2)=O)c[nH]c2cc(C#N)ccc12 N1(C(CCSC)=O)CCN(C(c2ccc(CN3CCCCC3C)cc2)=O)CC1C C(=O)(C1CCc2cccnc21)NC(C1N(C(CC(C)(C)OC)=O)CCC1)C N1(C(C2(CC=C)COC2)=O)CC2(CCCC2NC(c2cc(C(C)C)oc2C)=O)C1 N1(CC(=O)NC2(CNC(CCC3CCC(C)O3)=O)CCC2)CCC(O)CC1 C12(NC(c3occ(C)c3C)=O)CCC1CN(C(C1(F)CCS(=O)(=O)C1)=O)C2 N1(C(CCOCCCOC)=O)CCC(O)(CNC(c2cc(CN(C)C)c[nH]2)=O)C1 CC1(NC(C2CC2[N+](=O)[O-])=O)CCN(C(=O)CSCc2cccs2)CC1 N1(C(c2cnc(C)[nH]2)=O)CC2C(NC(=O)CC(C)N(C)C)CS(=O)(=O)C2C1 c1(NC(=O)OC)c[nH]c(Br)c1.C(=O)(C(CC)n1cccc1)NCCN(CC)CC C(C(C(C)(C)C)NC(c1cccc(OCC(C)C)c1)=O)NC(c1onc(C)n1)=O c1(C(=O)NCC2CCN(C(c3cn(CC)nn3)=O)C2)ccc(Br)cc1C C(=O)(CCCCC(C)=O)NC1CC=C(C(=O)NC(CCCC)C)C1 N1(C(C2(C)CC2(Cl)Cl)=O)CCc2[nH]nc(CNC(C3CC4C=CC3C4)=O)c2C1 N1(C(C2(CC)CCCN2C(=O)C=Cc2cocn2)=O)CC(CO)C(C)(C)C1 Cc1nc(N)cnc1C(=O)NC1C2CCC1N(C(C1(C)CCCS1)=O)C2 C(N=c1nc(N2CCOC(C)CC2)c2sccc2[nH]1)C1N(CC)CC1 C(=O)(C1=CS(=O)(=O)CCC1)NC1CCCC(NC(c2c(C)ncn2O)=O)CC1 N1(C(CSC)=O)CCC(C(=O)NC2CC23CCCC3)(OC)C1 C#CC1(C(N2CCC(CNC(C3(C)CC(C#N)C3)=O)C2)=O)CCCC1 N1(C(C2(C)C(C)CN(C(=O)CCCC3CC3)C2)=O)CCCC2(CCCC2)C1 N1(C(C2N(C(C(C)N(CC)CC)=O)CC2C)=O)CC2CCCCC2C1 C(=O)(C(CC(C)C)NC(=O)OC)N1CC(CNC(C(CC)C2CCOCC2)=O)C1 c1(-n2cc(CC(N3CCC(C(F)(F)F)(C(=O)O)C3)=O)nn2)ccc2c(c1)CCC2 CCC(C)CC(=O)NCC(CO)NC(c1csc(-c2csc(C)n2)c1)=O c1(C(c2ccn(C)n2)NCC2(OC)CC2)nnnn1CCSC Cc1cccn(CC(N2CCC(NC(C3(n4cccn4)CC3)=O)C2C)=O)c1=O C(CC(CCO)NC(=O)CC1COCCN1C(=O)Cn1ccc(C)c1)SC O=C(NNc1ccc2ccccc2n1)NCC1Cc2ccccc2CO1 C1(CC(C)C)CCCC1(C)NC(=O)CCCC1CC1C c1(SCC(=O)NCC(C)N(C(=O)CCSCCC(C)C)CC)csc(C)c1 C1(NC(c2cccc(C)c2F)=O)CC2(CCC(NC(C3(C)CCCO3)=O)CC2)C1 N1(C(C(CC)NC(N)=O)=O)CCCN(C(c2cccc(F)c2)=O)CC1C c1(N2CC(C(=O)NCC(COC)C)C2)nncn1C c1(CN2CC(NC(C3C(OCC)CCC3)=O)C(F)C2)cccc(Cl)c1O C(=O)(C(C)CC(F)F)NC1(C(=O)NCCCC)CCC1 C1(C(=O)NCC(C)CNC(=O)C=C2SCC(=O)N2C)CCc2cc(F)ccc2O1 C=C(C)C(C)(C)C(=O)N1CCN(C(=O)C(C)Cc2ccco2)C(CC(C)(C)C)C1 c1(NCC2CCC(NC(C3(C)CC3Br)=O)CC2)ccc([N+](=O)[O-])c2cccnc12 C1(NC(C(C2CN(C(C(C)OC)=O)C2)O)=O)CCCN(C2CC2)C1 c1(C(=O)NC2CN(C(c3c(COC)nn[nH]3)=O)C(C)(C)C2)cncc([N+](=O)[O-])c1 C1(C(F)(F)F)(C(N(CC(C)N(C(CN(CCC#C)C)=O)C)C)=O)CCCCC1 CCC(CC(=O)NC(C(=O)N(C1CN(C(C)C)C1)C)C1(C)CC1)OC C1(C)(CNC(C=C(C)Cl)=O)CN(C(=O)COCc2ncc(C)o2)CCO1 C1(CNC(=O)C=Cc2cnc[nH]2)CC12CCN(C(c1nnc(O)nc1O)=O)CC2 C(=O)(CC(F)(F)C(F)F)NC(CNC(=O)C#CC1CC1)C1CCC1 N1(C(C(C(C)(C)C)(C)C)=O)CCC2(CC1)CC(NC(=O)C#CC1CCCOC1)C2 N1(CC(=O)N(CCCNC(C2CCN(C)CC2)=O)C)CC(C(F)(F)F)CCC1=O c1(CC)cncc(C(=O)NC2CCCC(N(C(=O)Cc3cnc[nH]3)C)C2)c1 C(C(O)C(=O)N1CC(O)(CNC(C2(S(C)(=O)=O)CC2)=O)C1)N(C)C c1(CC)nc(C(=O)NCC(=O)NCC2C=CCOC2)co1 CC(C)C1=NOC(C)(C(=O)NCC2COCCN(C(=O)C(F)=C3CCC3)C2)C1 N1(C(C(CC)N(C)C)=O)CCCCC1CCCNC(=O)COCC(C)(C)C CCC1=NOC(CC(N2CC=CC(C(=O)N(C(C)C)CC)C2)=O)C1 C(=O)(CCP(C)(C)=O)NCC(CCOC)NC(c1cc(C(C)C)ccc1C)=O c1(C(N(CC(C)NC(=O)C2=CSCS2)CC)=O)cn2ccsc2n1 N1(C(=O)Nc2ccc(F)cc2)CCC2(CCC2)C(C(=O)C=CC2CCOC2)C1 c1(-c2nc(C)nn2Cc2cccc(C)c2C)cc(S(C)(=O)=O)c(Cl)cc1Cl C1(C)(NC(CN(C(c2c(C)scc2)=O)CC2CC2)=O)CCCC(C)(C)C1 c1(CC)ccccc1CC(=O)NCC1CCCCN1C(C1CC(=O)C1C)=O CN=c1ccc(C(=O)NCC2CCCCC2C(=O)N(C)Cc2nc(C)cs2)c[nH]1 N1(C(CCCCC)=O)CCCC(O)(CNC(c2cn(C3CCOC3)nn2)=O)CC1 n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N(C)CC2CCC(=O)N2)cc1C c1(C(=O)OC)ccc(NC(=O)Cc2cnn(C(C)C)c2)c2ncccc12 C(=O)(C(CC)(CC)CC)NC1C(C(=O)NC(CC)C2CC2)CC=CC1 N1(C(COC(C)C)=O)CC(O)CC1Cn1cc(SCCO)nn1 C12(C(=O)NCC3C4CN(C(=O)CC=Cc5ccccc5)CC34)COCC1C2(F)F Cc1cc(C(=O)NCC23CCC2CCN3C(C23CC(C)(C2)C3)=O)c(C)cn1 O=C(N=c1[nH]n(Cc2ccco2)cc1Br)c1snnc1C1CCC1 c1(C(=O)NCC2C(NC(c3ncn(CC)n3)=O)C2)cccc(Cl)c1N c1(NC)cnccc1C(=O)N(C1CN(C(=O)C(c2ccccc2F)OC)C1)C CCC(C)(CCO)NC(C1CN(C(=O)CN2CCC(F)CC2)CC1OC)=O N1(C(C2C(C)OCC2)=O)CCCCC(CNC(c2cc(C(F)F)cc(F)c2)=O)C1 N1(C(CN(C)CC)=O)CC2CC(C(=O)NC(C)C(C)(C)C(=O)NC)C(C2)C1 Cn1[nH]c(C(=O)NCC2CC(NC(=O)COc3cccc(O)c3)C2)nc1=O N1(C(C(C)=O)C)CCC(C(=O)N(CCOCCOCC)C(C)C)CC1.c1(O)nc[nH]n1 c1(C(N2C(C)C(NC(=O)CCC3CC3(F)F)CCC2)=O)ccc(C#N)c(Cl)c1 C1(NC(c2c(C(C)C)c[nH]n2)=O)CN(C(c2cc(C3CC3C)on2)=O)C(C)(C)C1 C(C)(C)(C(=O)NC1CN(C(=O)C(F)=CC2CC2)C1)N(C)C c1(C(N2CC3C(CNS(CC=C)(=O)=O)C3C2)=O)ccc(F)c(S(C)(=O)=O)c1 Cc1ccc(Br)nc1C(=O)NCCCn1cc(C(C)(C)C(N)=O)nn1 CCC(=O)CCC(=O)NCC1OCCC1C(=O)NCc1cccc(OC)n1 Cc1ccoc1CC(=O)Nc1nc(C2CCOC2)cs1 NC(=O)CC(O)C(=O)NC1CCCN(C(c2ccc(O)cc2Cl)=O)C1 CCS(=O)CC(=O)N1CCN(CC2CCCN(C(=O)Cn3ccnn3)C2)CC1 C(=O)(C(O)CC(F)(F)F)N1CCN(C(CCC=CCC=C)=O)C(CC(F)(F)F)C1 c1(C(N2CC(CNC(C(C)N(C)C)=O)C(C)C2)=O)cc(Br)c2n[nH]cc2c1 c1(C(=O)NCC2CC(C)N(C(=O)CC3(C)CC3(F)Cl)C2)cnc2c(ccn2C)c1 N1(C(c2c(C)c(Br)n(C)n2)=O)C2CCC1C(C)C(NC(c1ccoc1)=O)C2 C1(OCC)CC(Nc2ncccc2Br)C12CCOCC2 C=CCCCC(C)NC(=O)COC1CCN(C(c2n[nH]c(C)c2Cl)=O)C1 C1(OC)CC2CC(C1)N(C(=O)NC1CC3(CCCCC3)C1)C2 c1(C(C)C)ccc(N2CCOCC2)c(C#N)n1.C12CN(C3(CCOC3)C1)C2 C=CCCCCCC(=O)NCC=C1CCN(C(C2CC2(C(C)C)CC)=O)CC1 Cc1nn(C)cc1C(=O)N(CCNC(=O)CN(C)CCc1ccccc1)C1CC1 Cc1csc(CCC(=O)NCC2(C(C)(C)O)CN(C(c3cncnc3)=O)C2)n1 c1(C(C(=O)NCCN(C(C2COCCO2)=O)CC)C)ccc(C)cc1 C1(C(C)SCC)CCCN(C(=O)C(CCO)CCNC)C1.O(C(F)F)CCOCCO c1(C(=O)NCC(CC)NC(C(CC)SC)=O)c(C)nn(C)c1F c1(C(N(CCNC(c2ccncn2)=O)CC)=O)cc([N+](=O)[O-])ccc1N(C)C c1(C(=O)NC2C3CN(C(C(CCC)N4CCNCC4)=O)CC32)c(C)cccc1C Cc1ccncc1CC(=O)NCC1CC2CC2N1C(=O)C(F)CC1CC1 C=C(C)C(C)(O)C(=O)N1CCCC(CNC(c2sc(-c3ncc[nH]3)nc2C)=O)C1 c1(C(=O)NCC2(F)CC(NC(C(C)n3cncn3)=O)C2)cccc2c1CCN2 CCCC(CC)CCC(=O)NC12CCC(CC1)CC2.C1(=O)NOCCC12CC2 C(=O)(CCCC(F)F)N(C1CCCN(C(C2CCC23CCC3)=O)C1)CCO C1(CCNC(c2cc(N(C)C)ncc2)=O)CN(C(c2csc(Cl)c2)=O)CCCO1 c1(CC)cc(C(=O)NC2CN(C(C3C(C)C3C)=O)CC2c2cnn(C)c2)c(C)o1 C(c1ccc(C)c(C)c1)=CC(N1CCN(C(CSC)=O)C(c2ccnn2C)C1)=O C12(CNC(c3nc(C#C)sc3)=O)CC(CO1)N(C(=O)C(C)CC(C)C)C2 c1(C(=O)NC2CCCC2CNC(C2CC(F)(CO)C2)=O)cc(F)c(F)cc1O N1(C(C=C(COC)C)=O)CCC2(NC(c3cc(SC)oc3C)=O)CCCCCC12 c1(C(N2C(CNC(C(CC(C)C)OC)=O)CCC2)=O)cc2occ(Br)c2[nH]1 C1(CNC(=O)N(CC(C2CCCO2)O)CCO)CCS(=O)(=O)CC1 c1(CC)cnc(O)c(C(N2CCC(C)C2CNC(C2CCC(C)O2)=O)=O)c1 c1(C(N2C(C)(CNC(C(C(C)C)OC)=O)CCC2)=O)cccc([N+](=O)[O-])c1C Cc1csc(C(O)CC(=O)NCC(C)(C2CC2)NC(=O)OC(C)(C)C)c1 N1(C(c2cn(CC)nc2C(C)C)=O)CCCC12CCN(C(=O)CCS(C)=O)CC2 CC1(C)C(CNC(=O)CC2=CCCC2)CCN1C(c1ccc(N)c(Cl)c1)=O Cc1ccn(CC(=O)NC(Cn2cccn2)C(=O)NC(C)C(C)N(C)C)n1 N1(C(C(C)N2CCC2)=O)CCN(CCCCCNC(c2cocn2)=O)CC1 Cn1ncc(Cl)c1C(=O)NC1CC12CC(NC(=O)CCc1ccncn1)C2 C1(NC(C(C)OCCOCC)=O)CC2CCC1N2C(=O)CCC1CC1(Cl)Cl c1(C(N2C(C(C)NC(C3C(C)(C)C3(F)F)=O)CCC2)=O)nc2cccccc-2n1 c1(C(=O)NCCN2CCN(C(c3c[nH]c(=NC)o3)=O)CC2)cccc2c1CCC2 CCCC(C)(CC)C(=O)N(CCCNC(=O)C(C(C)C)n1cnnc1)CC C(c1ccc(F)cc1)=CC1CN(C(=O)CCn2cnnn2)C1 c1(C(=O)NCC(CNC(c2ccc(C)c(N)c2)=O)C)cccc2oncc12 C(=O)(CC(O)C(C)C)N1C(CNC(CCCn2c(C)cc(C)n2)=O)C=CC1 N1(C(=O)OC(C)(C)C)CCC(NC(=O)CCc2cccnc2)C(O)C1 C1(CNC(c2nnc(C)s2)=O)CC(C)N(C(c2nccc(C(F)(F)F)n2)=O)C1 c1(C(=O)NC(CNC(CC#N)=O)NC(C2CC2F)=O)ccccc1 CCCCC(O)C(C)C(=O)NCCCC(CO)NC(=O)CC1(CSC)CC1 Cc1ccc(C(=O)NCC2CN(C(=O)CC3C=CCCC3)CC2C)c(N)n1 CCC(CC(=O)N(CCCCCCNC(C1(C)CC1(F)F)=O)C)C1CCC1 N1(C(C(C)CO)=O)C(CNC(c2cc3cccn3cn2)=O)CC2CCCC12 C(=O)(C(C(C)(C)C)N1CCC(CC2CCC2)C1)NCC(=O)OC(C)(C)C C(=O)(C(CNC(=O)C=Cc1cc[nH]n1)N(C)C)N(C(c1ccco1)C)C C1(C(C)(C)NC(=O)CC2CCCC2)CCCN1C(c1cnn(CC(F)F)n1)=O C1(N(C(c2c(CCC)nco2)=O)C)CCCC(NC(C2(C(C)C)CCC2)=O)C1 C(=O)(C(CC(N)=O)NC(c1ccnc(C)n1)=O)N1CCCC(CCC#C)C1 c1(OC)cc(NC(C2CCN2CC2CCOC2(C)C)=O)ccc1C Cc1c(C(=O)NCC(C)(C)OCC(=O)NCc2nn(C)cc2C)[nH]ccc1=O CCCCCCC(CC)(CC)C(=O)N1CC(NC(C2CS(=O)(=O)CC(=O)N2)=O)C1 C(=O)(C(CC(C)(C)C)OC)NC1C(CC(=O)NCCN(CCO)CC)CCC1 CC(C)C(C#N)C(=O)NCC1CCN1C(c1ccnn1C(C)(C)C)=O C1(NC(C2CCCO2)=O)CN(C(=O)C(F)=CCCF)CC12CCCC2 C1(C(C)(C)C)(CO)CCN(C(=O)CC2CC2)CC1.C(=O)(CC1CCO1)N c1(C(N2CC(NC(c3cc(C)nn3C)=O)CC2(C)C)=O)ccc2nccn2n1 CC(C)C(C(=O)NC1CCC1C(N1CCOC(C(N)=O)C1)=O)C(C)C C1(C)(NC(C2N(S(C)(=O)=O)CCC2)=O)CCN(C(C23CC(CO2)C3)=O)C1 C(=O)(C1CCCc2c(O)cccc21)N1CC(C)(NC(C2CC3CCC2CC3)=O)C1 C(=O)(C1=C(C(C)CC)N(Cc2ccc(Cl)s2)C(=S)NC1c1cocn1)OCC c1(C(=O)NCC(CNC(=O)CC2CC(n3cccn3)C2)CO)cc(F)cc(Cl)c1 c1(C(N2C3CCC2CC(NC(C24CCC2C4)=O)C3)=O)c[nH]c(=O)c2ccncc12 C1(NC(C2ON=C(C)C2)=O)CC2CC(C1)CN(C(c1nn(C)cc1[N+](=O)[O-])=O)C2 C(=O)(C(C)CC(F)F)N1CCC(N2CCC(NC(c3cnc(C)[nH]3)=O)CC2)C1 Cc1cccc(NC(=O)C(N2CCC(CN(C)C(c3c[nH]cc3Br)=O)C2)=O)c1C c1(CCNC2=NCC3C(C)(C3)CN2)nc2ncccn2n1.C(F)(F)F N1(C(C(C(C)O)C)=O)CC2CC(C)N(C(c3cccc(NC(N)=O)c3)=O)C2C1 c1(C(=O)NCC(CNC(c2c(C)ccs2)=O)(C)C)ccc(F)c(C)c1N N1(C(C(CC(C)C)O)=O)CCC2CCC(C1)N2C(=O)CCCNC(c1cccs1)=O N1(C(c2c(C)cns2)=O)CCC(C)(C)CC1C(N1CC2CC2(CO)C1)=O c1(N(CCCCSC)C)nc2c(c(=NCc3ccc(C4CC4)o3)[nH]1)CC(C)CC2 CCC(C)CC(=O)NC1CCN(C(c2ccn(C)n2)=O)C1C CC1(C)CC(NC(c2cc(C(N)=O)co2)=O)CCN(C(=O)C=CBr)C1 c1(CCC(=O)NC(CCCC)CNC(c2snnc2C)=O)ccc(OC)cc1F N1(C(C2CCC(CNC(=O)CCc3nccs3)C2)=O)CCC(CC(N)=O)CC1 c1(CNC(=O)NC2CCCC2CF)c(Cl)cc(Cl)cc1Cl Cc1ccc(CC(=O)N(CCNC(c2ncc(N)cc2C)=O)C2CC2)c(C)c1 C1(NC(c2ccc(N)c(F)n2)=O)CCN(C(c2cccc(Cl)c2)=O)CCC1(F)F c1(OCC(C)C)ccc(Cl)c(C(=O)NC2CCC(C)(CNC(C3CSC3)=O)C2)n1 C1(CCC(=O)NCCCCOC)CCCCN1C(=O)C(c1cccnc1)C N1(C(CCC2N(C)CCC2)=O)CCCC(C)(CNC(c2ccccn2)=O)C1 N1(C(C2CCCC(=O)C2)=O)CCCCCC1C(=O)NC1CCCSCC1 S(=O)(=O)(c1ccc(Br)c2ccccc12)NC(C(=O)OC)C(C)C1CC1 N1(C(=O)NC(C(=O)OC)C)CC(C)(C)Oc2ccc(NC3CCCCC3)cc21 c1(NC(Cc2cc(C(=O)OC)c(Br)cc2)=O)cnn2c1OCC(O)C2 CCCCCCC(C)NC(c1cc(CNC(C2(COCC)CC2)=O)no1)=O CC1(C)CCC(CC(N2CCCC2C(O)CO)=O)OC1 C=C(Cl)CCC(=O)NCC1C=CCN1C(c1cccc(C(C)(F)F)c1)=O C1(CC(N2CC(NC(C(C=C=C)C)=O)C(SC)C2)=O)CCN(OC)CC1 C(=O)(CCCCC(N)=O)NC1(CCNC(c2c(C)cccc2F)=O)CC1 C(CN=S(C)(C)=O)NC(C(CO)NC(C(CC)n1ccnc1)=O)=O C1(C(C(=O)NCSc2ccccc2O)N(C2CCOC2)C)CC2(C1)OCCO2 c1(C(N(CCNC(c2cccc(CC)c2)=O)C)=O)ccnc(S(N)(=O)=O)c1 N1(C(C2CCC(CNC(C(C#N)C3CC3)=O)O2)=O)CC(O)C(O)C1 CC(CC(=O)NCC(C1CCCC1)NC(c1cnc(C(C)(C)C)o1)=O)N(C)C Cc1nn(CC(N2CCOCC2CNC(C2(CF)CCOCC2)=O)=O)cc1Cl C12(CC)CCC(C(=O)NCC3CCC(NC(=O)CNS(=O)(=O)N(C)C)C3)(CO1)C2 N1(C(C2(N)CCCC2)C(=O)OC)CCc2[nH]c3ccc(F)cc3c2C1.O(C)CC C(C1CCCN1C)=CC(=O)NCC(=CC(N1CCC(NC(=O)NC)C1)=O)C c1(C(=O)NCCC(C)NC(=O)CCCCC(F)F)cn(C)c(=O)c2c1CCCC2 C(=O)(C(C)(C)CCCC(=O)N1CC2CC2(NC(c2cnnc(O)c2)=O)C1)OC C(=O)(CCCCCOCC)N1CC(NC(C=CC)=O)C(SC)C1 Cc1cc(C(=O)NCCCC(C)NC(c2ccnn2C2CCCC2)=O)cc(N)c1 N12CCOC(CC1)C2=O.c1(NC)cnccc1C(N1CC=CC(OC)C1)=O N1(C(C2(OC)CCC2)=O)CCC(CO)(CNC(=O)CC2CCCCC23CC3)CC1 c1(C(N2CCN(C(C(CC=C)CC)=O)C(CCOC)C2)=O)cc(C#N)ccc1C C1(CNC2(CO)CCN(CC)C2)CC2(C1)CC1(CC(C(=O)O)C1)C2 CCC(C(=O)N(CCCNC(c1cc(CC(C)C)[nH]n1)=O)CC1CCCC1)OC N1(C(C2CCC(C)C2)=O)CCC(C2CN(C(c3ccsc3Cl)=O)C2)CC1 c1(C(N2CC(C#N)C(NC(c3cc(Cl)ccn3)=O)C2)=O)ccc2scnc2c1 S(=O)(=O)(c1cncc(Br)c1)N1CC(C(=O)Nc2cc(F)c(Cl)cn2)C(F)(F)CC1 c1(NC(CC=C)(C)C)ccc(S(=O)(=O)N2CCC(C3CCN(C)C3)C2)cc1F CC1CN(C(=O)CC(CNC(C2(C)CC2(C)C)=O)C2CCC2)CC1O c1(C(=O)NC2C(C)CN(C(=O)C=Cc3ncco3)C2)cc(O)nc(O)c1 Cc1cc(C(=O)NCC2(O)CCN(C(=O)CCc3cncn3C)C2)c(C)s1 C(=O)(CC(C)CC(F)(F)F)NCCC1(NC(Cn2c(C)c(Cl)cn2)=O)CCCC1 C(=O)(C1=NN=C(NCc2cnc3n2CCCC3)OCC1)OCC c1(C(=O)NC2CC(C(=O)NCc3ccccc3C3CC3)C2)ccc(F)cc1O c1(C(C)C)nn(C)cc1C(N1CC(NC(=O)Cc2cnc[nH]2)C(O)C1)=O C1(C(C)C)(C(=O)NC2CC2CNC(=O)Cn2cnc([N+](=O)[O-])n2)CCN(C)CC1 c1(CC(=O)OCCC(=O)NC(COCC)(C)C(=O)O)ccccc1CC C(=O)(CCC(=O)NCC(CO)NC(C1CCCN1CC(C)C)=O)OCC CCCC(O)CC(=O)NCC1CC(F)(CNC(c2sccc2SC(F)F)=O)C1 c1(C(c2nnnn2C2CCC2)(F)NC(CC)COC(C)C)ccc(C#N)cc1 n1(CC)c(C(C)NC(=O)CC2(C)CCOC2)nc2ccccc12 c1(CN(CCOC)C)nc(-c2c[nH]nc2Cl)n(C2CCC2)n1 CCCCCC(F)C(=O)NC1CN(C(=O)C(c2cnn(C)c2)OC)CCC12CC2 N1(C(c2cc(C)sc2C)C(=O)NCC=C)CCCSCC1C c1(OC)cc(C(=O)NC(C)CCCNC(=O)Cc2cn(C)nn2)c(C)cc1O CC1CCOC(C(N2CC(N3CCN(C(=O)C4=COCC4)CC3)C2)=O)C1 C1(CCNC(c2ccc(OC)o2)=O)CN(C(C2(CC(F)F)CC2)=O)CC1C C1(CNC(CCc2nc(C)sc2)=O)CCN(C(C2CCCC2)=O)C(C)C1 N1(C(C(c2c[nH]c(=N)s2)C)=O)CCC2C(CCCN2C(=O)CCc2ccccn2)C1 C(CCC(=O)NCCc1cccc(O)n1)(C(C)C)NC(C(CC#C)(C)C)=O CCCCS(=O)(=O)CC(=O)OC1CC2(CCC2NC(=O)OC(C)(C)C)C1 N(C(=NCCc1ccoc1)N1CCCC(CC(N)=O)C1)C1CC(O)C1 C1(NC(C=CSC)=O)CCC2(CCN(C(c3ccc(Cl)c([N+](=O)[O-])c3)=O)CC2)C1 c1(OC)ccc(C(C)(C)C(=O)N(CC(O)CNC(=O)CC(C)C2CC2)C)cc1 c1(CC(C)C)ccc(CO)cn1.c12ccc(cn1)C(=O)NCC(C)n1cc-2nn1 N1(C(c2n(CC)cc(Cl)c2)=O)CCC(N(C)C(c2ccc(C)c(Cl)c2)=O)C(C)C1 C=CC(C)(C)CC(=O)NCc1cc(C(=O)NC(C)C(C)C)cs1 C1(CCC)C(=O)NCCN1C(=O)C(C)(C)C(C)NC(c1nnn(C)c1C)=O c1(OC)cc(C)cc(C(=O)NCC(C2CC2)NC(c2ccnnc2)=O)c1O c1(CNC2CCN(C(c3nc(C)sc3)=O)CC2O)n[nH]c2ccc(Cl)cc12 C(CCC(CCC)NC(=O)Cc1cnsc1)NC(CC(C=C)C)=O CCCCC(C)N=c1nc(N(CC(F)(F)Cl)C)c2ccc(N3CCOCC3)cc2[nH]1 c1(CC(N2CC(CN(C(=O)C(C)NC(C)(C)C)C)C2)=O)cnc(C)[nH]1 C1(NCc2c(Br)ncnc2Cl)CC2CCC(C1)N2S(=O)(=O)c1cccnc1 CCC(COC)C(=O)NC(C)(C)CCNC(=O)C(C)NC(c1ccoc1)=O CCCCCCC(C)C(=O)NCC1C(C)CCN1C(C1CCC1)=O c1(C(N2CCC3(NC(COC)=O)C(C2)C3)=O)cnc2c(c1)CNC2=O Cn1c2c(ccc1=O)C(NC(C1(C)CCC(C)(C)CC1)=O)CCC2 C1(NC(c2ccc(SC(F)(F)F)cc2)=O)CCCCN(C(c2csc(Cl)c2)=O)C1 O=C1Cc2ccc(C(N3CC=CC3CNC(=O)C(F)CC3CCC3)=O)cc2N1 c1(Oc2ccc(NC(CNC(C(C)(C)CO)=O)=O)cn2)cc(Br)ccc1F N1(C(C(COC)C)=O)CC(OC)C(C(=O)NCc2cccc(OC(F)F)c2)C1 CC12CC3CC(CC(C(=O)NCC4CCCCN4C(c4cccnc4)=O)(C3)C1)C2 N1(C(C(CCCC)O)=O)CCC(C(=O)NCc2cc(F)cc(F)c2)=C(F)C1 c1(C(=O)NC(CNC(CN(CCCCCC)C)=O)C)ccc(Br)c(C)n1 N1(C(C2CN(C)C(=O)N2)=O)CC(=O)NCC1C(=O)Nc1cnn(CC(N)=O)c1 Cc1cc(C(=O)NC2CCC(NC(=O)C(C)OC3CCCCC3)C2)sn1 S(=O)(=O)(c1cc(C)c(Cl)c(C)c1)N1C(C)CCC(CC)C1 CC1(C)CN(C(C2(C)CC=CCO2)=O)CC(CNC(=O)CCF)O1 C(=O)(C1=CC(C)CC1)N1CCC(C(N)=O)(NC)C1 c1(OC)ccc(Cl)c(C(N2CC3(CCN3C(c3cnc[nH]3)=O)C2)=O)c1N c1(C(=O)NC2CN(C(C3C(C)(COC)C3)=O)CC2(C)C)coc2ccccc12 C12(CNC(CSC)=O)CCCCC1N(C(c1cc(F)c(C(F)F)cc1F)=O)CC2 Cc1cc(CCCCN(S(=O)(=O)CCOCC(C)C)CC)cc(C)n1.C1CCOCC1 N1(C(c2nc(C)sc2Br)=O)CCC2(CCCCC2NC(C2CC23CCC3)=O)C1 C1(COC)(CNC(C2(C)CCOC2)=O)CCCN1C(c1cccnc1S)=O C(=O)(CC(O)C(C)C)NCC(C)NC(=O)Cc1ccc(-n2cnnn2)cc1 C1(NC(C2CCN(C)C2)=O)(CF)CCN(C(=O)C=Cc2ncc[nH]2)C1 N1(C(CNOC2CCCC(C)C2)=O)C2CCC(C2)C1CC(=O)NCCC(C(=C)C)=O c1(C(N(CCCCNC(=O)CC2NC(=O)NC2=O)C)=O)ccn(CCO)c(=O)c1 c1(C(=O)NCCCC2(NC(c3cnc(O)o3)=O)CC2)cccc2[nH]ccc12 Cc1cccc(C(N2CCC(O)(CNC(=O)CCC3CCN(C)CC3)C2)=O)c1O N1(C(C2N(C(C)=O)CCC2)=O)CCC2CN(Cc3c(C)nn(C)c3Cl)CC12 c1(C(=O)NC(C)C(C)NC(=O)CCc2cn[nH]c2)ccnc(N(C)C)c1 N1(c2n(CC3(COC)CC3)nnn2)CCc2c(F)ccc(Br)c2C1 c1(OCC)ccc(C(C)Nc2cccc(-c3nc(C)cs3)c2)cc1OC C1(OCC)(CNC(=O)CCN(CCCO)C(c2[nH]nnc2C)=O)CCCCC1 c1(NC(c2c(CNC(Cc3ccc(C)s3)=O)cco2)=O)ccc[n+]([O-])c1 c1(-c2ccc(OC)s2)cccc2c(C(N3CCC(OC)CC3)=O)[nH]nc12 c1(C(N2CCCCC(CNC(C3CC(O)C3)=O)C2)=O)ccc2ccc(Cl)cc2n1 c1(N)ccc2occc2c1.c1(C(C)Cc2nnnn2C(C)C)cnn(C(C)(C)C)c1 c1(CC(C)C(=O)NC2CC2CNC(=O)CC(C)(C)C)cccc(F)c1 c1(CC)ccc(OC)c(CN2CCCC2C(N2CCCC(O)C2C)=O)c1 c1(C(N2CCCC(NC(C3CN(CC)C(=O)C3)=O)C2)=O)ccc2c(c1)CC2 N1(C(CCC=C)=O)CCC(C)N(C(C2CCOC(CC)C2)=O)CC1 C1(C(=O)OC(C(C)NC(=O)OC(C)(C)C)=O)CCCN1c1ccncn1.C1(CO)CC1F N1(C(C(CC)(C)C)=O)CCC(CNC(c2cccc(C)c2)=O)C(F)(F)CC1 CC1CC(CC(=O)NCc2cn(C3CC3)cn2)CN1C(C1CCC1)=O C(=O)(C(C)(C)CS(N)(=O)=O)N(CC(C)N(C(C=Cc1ncc(C)[nH]1)=O)C)C C1(NC(C(C)CF)=O)COC2(C1)CN(C(c1cc(Cl)ncc1N)=O)C2 C1(CC(NC(=S)Nc2cccc(Br)c2)=O)Oc2ccccc2NC1=O C1(C(=O)Nc2cn(CC(C)C)nc2)C2CC2CN1C(C1CCC1(F)F)=O Cc1c(C(=O)NCCC(O)CNC(c2c[nH]nc2C2CCC2)=O)cnn1C(C)C C(CN=c1cc(C)c(S(=O)(=O)NC2CN(C)CC2OC)c[nH]1)N(CC)CC C12(C(=O)NCc3ccc(OC)nn3)CCC(CC1NC(c1cn(C)nc1C)=O)C2 C1(CC)CN(C(c2cc(CO)[nH]n2)=O)CC1C(=O)NCC1(C)CCCCO1 c1(NC(C2CN(C(C(=O)NC(C)C)=O)CC2C)=O)cccc(C2CC2)c1Cl c1(C(N(C2CCOC2)C)=O)ccc([Si](C)(C)C)cc1 CC(C)CC(CC(=O)N1CCCNC(=O)CC1)NC(C1C=CCS1)=O Cc1nn(CC(=O)NCC(CO)NC(=O)CN2CCC(O)CC2)c(C)c1Br c1(C(N2C(C)CN(Cc3nnn(C)n3)CC2)=O)ccc2cc[nH]c2n1 N1(C(C2CC(C)C2)=O)CC=CCC1C(=O)NC(CO)C1CCC1 C12(CC(=O)NCC(CNC(Cc3c(C)n(C)nc3)=O)CO)CCCN1CCC2 C(=O)(C(C)CCC(C)(C)C)NCC1OCCN(C(c2c(C)cc[nH]c2=N)=O)C1 C1(C(=O)NC(C=C)CO)CCOCCN1C(=O)Cc1nocc1C C(=O)(C1=CC2CC(C1)CC2O)N1CC(OC)C(NC(C2COC2)=O)C1 N1(C(C)=O)CCOCC2(CC(CNC(C3CC3(F)Cl)=O)CO2)C1 C1(C(=O)NC2C(OC(C)C)CCC2)C2CC1N(C(C1CCCC(CF)C1)=O)C2 C1(C(=O)NCC2C(=C)CC2)CCC(C)N(C(n2nc(C)cc2C(=O)O)=O)C1 CC1(CNC(=O)CCN(C(=O)CC2OCCCO2)C2CC2)COCCO1 CCC(C)(C)C(=O)C(=O)N1CCC(C2(NC(=O)C=Cc3cncc(F)c3)CC2)C1 CN1CC2(CCN2C(C2C(NC(=O)CCc3ccncn3)CCSC2)=O)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(C)(CNC(c2c(CC)cccc2)=O)C1 N1(C(C(CC)n2ccc(CC)n2)=O)CCC(NC(=O)Cc2n[nH]c(C)n2)CC1C c1(CC)cc(C(=O)N(C(C)C(=O)NCC2C=CCOC2)C2CC2)no1 C1(C(=O)NCC2C(CN(C(=O)CC(C)(C)N(C)C)C)CCC2)CC12CC2(F)F c1(C=O)oc(CC2CCCN2C(=O)CN(CCCCC)C2CC2)cc1C.OC N1(C(Cn2cc(CCOCC(=O)NCC)nn2)=O)CC2(COC(=O)C2)C1 C1CCCC1.O=C(C=CC1CC1)NCCOCCNC(C1CC1Cl)=O N1(C(C(=O)N(CC)CC)=O)CCC(C)CC1.c12cc(on1)C(=O)N2 CC1(CNC(C2(C#N)CCCO2)=O)CCN(C(=O)CCC(=O)C2CCCCC2)C1 N1(C(c2n(CC)ncc2Cl)=O)CCCC(CNC(=O)CN2CC3CC3C2)CC1 N1(C(C2(CC)CC2(F)F)=O)CC2CN(C(c3ccc4nnnn4c3)=O)CC2(C)C1 c1(OC)cc(-c2cnccc2C(=O)Nc2cnnc(OC)c2)c(OC)nn1 c1(C(N2CC(F)(CNC(C(CC)OC)=O)C2)=O)cc(S(N)(=O)=O)ccn1 c1(CC(=O)NC2(CNC(=O)Cn3nccn3)COC2)cccc(Br)c1 C12(F)CCN(CC1)C2.c1(OC)cccc(CNC(C2CN(C)C2)=O)n1 Cc1cc(C(=O)NC2CCC(CNC(c3ccc(C4CC4)s3)=O)CC2)ccn1 N1(CC(N2CC(CNC(=O)CO)C2)=O)CCCCS1(=O)=O C1(C(N2C(C)CC(F)C2)=O)CN(C(C2CCC(C)(C)OC2)=O)CC1(C)C c1(CC(=O)NCC2(F)CCC(NC(C3C(CC)CCC3)=O)C2)ccc(F)c(F)c1 C12(SCC)CN(C(C)=O)C(CNC(=O)NC(C3CC3)N(C)C)(C1)C2 c1(C(N2CC(NC(C=CC(C)(C)C)=O)C(F)C2)=O)c[nH]c2c(Cl)cccc12 c1(NC(c2n(CCC)nnn2)c2ccc(C)o2)ccc(Br)c2c1CCCC2 Cn1nc(Cl)cc1C(=O)NCC1(C)CCN(C(C2(CO)CCC2)=O)C1 CC1CCOCC1C(=O)NC12CC1CN(C(C1(OC(C)C)CCCC1)=O)C2 N1(C(c2ccc(OC(C)C)cc2O)=O)CCN(C(=O)CC(C)CF)CC2(CC2)C1 C(CC(C(=O)NCC1CCN(C(C2CCC(=O)NC2)=O)CC1)NC(C)=O)OC CP(C)(=O)C1CCCC1CNC(C1CCN(c2ccc(C(N)=O)cn2)CC1)=O c1(C(c2n(C(C)C)nnn2)NCC2(CCCl)CCC2)cccc(CO)c1 c1(C(=O)NC2C(NC(C3C(C=C)C3)=O)CC2)ccnc(CN(CC)CC)c1 C=CCC(C)(CC)C(=O)N1CC2CC(C(=O)NC3(C(N)=O)CCC3)C(C2)C1 c1(C(N2CC(CNC(c3c(C)n(C)nc3)=O)C(C)C2)=O)cc(O)nc(C2CC2)n1 c1(C(=O)NC2C(NC(=O)COCC3CCCC3)CCC2)cc(O)cc(F)c1 c1(C(=O)NC2C3CCN(C(C4(C5CC5)CCCO4)=O)CC23)cc2ncccn2n1 C1(C(=O)N(CC(=O)NC23CC(CNC(C(F)=CC)=O)(C2)C3)C)CCCCC1NC Cn1nccc(C(=O)NCC(CO)NC(C2(C)CS(=O)(=O)C2)=O)c1=O c1(NC2CC(=O)NC2)ncnc2c1ncn2Cc1ccc(OCC2CC2)cc1 C1(NC(COC)=O)CCN(Cc2sc(C)nc2Br)CC1 C1(O)(CC(=O)N(CCOCCNC(C2C(OC)CC2)=O)C)CCCCC1 n1(CC#C)ccc(C(=O)NCC2CCC(NC(=O)COCC(=C)C)C2)n1 O=C(CCC1CCc2ccccc21)NCC12CC1CN(C(c1cocn1)=O)C2 N1(C(=O)NCC(=O)Nc2c(OC)cccc2)CCC2CCCN(C(C)=O)C2C1 n1(CCC=C(C)C)cc(C2CCCN2C(=O)C(CC)N(c2ccccc2)C)nn1 N1(C(C2CC(C#C)(O)C2)=O)CCC(CNC(=O)C(COC)COC)C(F)(F)C1 c1(NC2CCC(SC)C2)ncnc(NC(C2CC(O)C2)C2CCCC2)c1C C1(C(N2C(C)COCC2)=O)C2C3CC4C1C2C34C(N(C)Cc1ccc(Cl)cc1)=O c1(OC)cccc(CC(=O)NC(CNC(=O)CO)CO)c1.C(=O)(C(O)C(C)C)NCC C(c1ccc(SC(F)F)cc1)=CC(=O)N(CC(C)NC(C1CCN(C)CC1)=O)C CC(=O)C(C)CC(C)C(=O)N1CCC1C(=O)NCC(C)(O)C1CCC1 C1(C(C)C)(C(=O)N(C)CC2OCCC2(C)C)CCCN1C(C1CN2CCC1C2)=O c1(OC)nc(OC)ccc1-c1cnn(C(C)=O)c1C C(CC(C)(C)C(=O)N(C1(CCO)CC1)C)NC(C(C)OC)=O C(=O)(CC(=O)NC(CC1CCCC1)C(=O)NC1CC1(C)C)NCC CCC(C)CCC(=O)N1CCCC(O)(CCNC(=O)Cc2cnn(C)c2)C1 c1(CC)ccc(C(=O)NCCC2CCC(NC(=O)CCCNC(=O)OC)C2)s1 CN1CC(C)(C)CC1C(N1CCC(Cn2cc(-c3ccc(C(=O)O)s3)nn2)C1)=O C=C1CC2(C1)CC(C(=O)NCC(O)CNC(c1cnc(OC)cc1C)=O)C2 c1(C(=O)NCC(CCOC)NC(C2CCN(C)C2)=O)cc(C(F)(F)F)ccc1Cl c1(C(N(CCC)CCNC(C2(O)CC2)=O)=O)cc(CC)cnc1O CN1CCCC(NC(C2CCN(C(=O)CC3CC=CCC3)CC2)=O)C1=O N1(C(C2CC(CCC)C2)=O)CCOC(CCCNC(c2cc(C)[nH]n2)=O)C1 c1(NC(=O)NC(C)C(=O)OC(=O)CC2CCC(=O)N2)ccccc1-n1cccn1 N1(C(CCNS(CC)(=O)=O)=O)CC2CC1C2NC(c1cnn(C(C)C)c1C)=O c1(N(c2cccnc2)CC(=C)Br)ncccc1S(=O)(=O)NC1CC(C#N)C1 Cc1cc(C(=O)NC2CCC(NC(=O)CCc3csc(=N)[nH]3)C2)c(C)n1C(C)C c1(C(=O)NC(C)CC2CCN(C(=O)CO)CC2)ccc2c(c1)NCC2 C(CCCC(=O)N(CC(C)(C)CNC(=O)CCC(C)N(C)C)CC)OCC CN1CCC2(CCN(C(=O)CC3CC(C)(C)CN3C(=O)CCC3CCCC3)C2)C1 C1(CC(=O)NCC(CCC)NC(C2CCN(OC)CC2)=O)CC(=O)NC(=O)C1 C(CS(=O)C(F)(F)F)NC(CC1C(c2ccc(OC)cc2)C1)=O c1(C(N2CCC(N(C)C(C3CCC4(CC4)C3)=O)CC2)=O)ccn2c(O)nnc2c1 C1(C(=O)NC(C)(C)CC=CC(=O)NCCN2CCCC(O)C2)CCCC(F)C1 N1(C(CCCOCCC)=O)CC2CC2(CNC(=O)CC2CCNC(=O)C2)C1 c1(C(N2CC(NC(c3cnc(CCC)s3)=O)C2)=O)ccc2c(c1)CCCO2 c1(C(N2CC(C(N3CC(C)CC(CC)C3)=O)C(OC)C2)=O)cc2cccnn2c1 Cc1nc(CCC(N2CCC(CO)(NC(c3ncoc3C)=O)C2)=O)oc1C C1(CNC(C(c2ccncc2)C)=O)CC(N=c2cc[nH]cc2C#N)C1 c1(C(N2CC(CNC(C(CN(C)C)(F)F)=O)C(O)C2)=O)cc(Cl)ccc1O C(=O)(CCS(N)(=O)=O)NCCCCCCN(C)C(C1CC1(F)Cl)=O N1(C(c2coc(C3CC3)c2)C(=O)NCc2cccs2)CCCC2CCC(O)CC12 Cc1c(CC(=O)NCC2(F)CCC(CNC(=O)C(C)O)C2)cccc1Br CCC(C)CCC(=O)NCC(CNC(=O)CSc1nncn1C1CC1)OC N1(C(C2CC(C)N(C(=O)Cn3ccnc3)CC2)=O)CCCNC(=O)C1C N1(C(C2C(C)(C(C)C)C2)=O)C2CCC1C(CNC(=O)C(C)n1cncn1)C2 C1(CNC(c2ccc(F)s2)=O)CN(C(=O)C(F)CC2CCOC2)C2(CCC2)C1 Cc1cnc(C(=O)NCCC2CCC(NC(c3cnoc3CC(C)C)=O)C2)cn1 C1(CC(=O)N(CCNC(c2cc(COC)sc2)=O)C2CC2)CCCC1(F)F N1(C(C2C(C)(C)C2)=O)CCC2CCC(NC(=O)CC=CCc3ccccc3)C12 C1(NC(c2cn(CCO)nn2)=O)(CO)CN(C(=O)C(F)(F)c2nccs2)C1 N1(C(C(CCC2CC2)NC(C(COCC)C)=O)=O)CCC(F)(F)C(F)C1 C1(CNC(C(CC=C)N(C)C)=O)CC2(C1)CN(C(=O)CCCCCC)C2 CCC(C)C(CN(C)C)NC(=O)CCn1cc(C(C)(C)CO)nn1 N1(C(c2[nH]c(=N)sc2)=O)CCCN(C(c2cccc3cncn23)=O)CCC1 Cc1c(C(=O)NCC2CCC(CNC(=O)C(C)(C)CC3CC3)CC2)cnn1C CN1CCC(O)(CNC(=O)COCCNC(C2CCOC2)=O)CC1 C12(C(N3CC(C)(C#N)C3)=O)CCCC1CN(C(=O)CCC(=O)C1CC1)C2 c1(C(=O)NC(CNC(C=CC=CCCCCC)=O)(C)C)cc(F)cc2cnccc12 C1(C(N2CC(F)(CNC(CN3CCN(CC)CC3)=O)C2)=O)CC(O)C12CCC2 c1(C(NOCC(N2CC3C(N(C)C)C3C2)=O)=O)ccc(C#N)cc1Br CCC(CNC(=O)CC1CC2(CCC2)C1)(CC)C(=O)N1CCC(F)C1 C(=O)(CC(C)(C)C(F)F)N(CCCCCNC(Cc1cccc(OC)c1)=O)C N1(C(CC)=O)CC2C(CNC(=O)CNC(=O)CCc3ccccn3)C2C1 c1(CN2CCCC(N(C3CN(C)CCO3)CC)C2)cc2c(s1)COCC2 c1(NC(C(N2CCCCC(C)C2)C=C)=O)c(C)cccc1C C1(C(=O)N(CC(=O)NCC#CCOC)CC2CC2)C2(CC2)C12CC2 N1(C(C2(c3cc(C)no3)CC2)=O)CCN(C(=O)C(C)c2cccs2)CC1C1CC1 N(C(=N)N1CC(O)CC(C)(C)C1)c1nn(C)c(Cl)c1[N+](=O)[O-] C=CCCCCCCC(=O)NCC1(F)CC(NC(=O)CC(=C)C)C1 C(=O)(C1=CN(CC(C)(C)C)CCC1)N1CC2C(NC(CSCCCC)=O)C(C2)C1 N1(C(CN(C)C)=O)CCN(c2nnc(C(c3cnccn3)C)n2CC2CC2)CC1 c1(CC(=O)NCCCC(C)(C)NC(C(CCCC)O)=O)ccc(S(C)=O)cc1 N1(C(C(C)(C(C)C)OC)=O)C2CC=C(C(=O)N(CC(C)O)CCO)C1CC2 C1(C(N2CC(NC(C3C4CCCC34)=O)CC(C)(C)C2)=O)Cc2cc(F)ccc2O1 C(C)(CCC(=O)NCCN1CCC(NC(C2C(C)C2(F)F)=O)CC1)OCC C(=O)(C(F)CC(C)C)N1C(CC)C(NC(=O)COC(C)(C)C)CC1 c1(NC(CCC=C)c2nnnn2C(C)(C)C)ccc(Cl)c(OC)c1 N(C1CCCc2ccoc21)C(c1n(CCOC)nnn1)c1cnn(CC(C)C)c1 CC1(C)CC(C(=O)NCCCCCCN(C)C)CCN1C(c1cc(C(N)=O)on1)=O N1(CCC)CCCC1CNC(=O)CN(C(C1CS(=O)C1)=O)C(C)C CC1CN(C(=O)CCSCC(N)=O)CC1NC(C1CCC(=O)C1)=O C1(NC(CNC(CC)=O)=O)(CC)CN(C(=O)C(c2ccccc2)O)C1 CC(C)C(CCNC(=O)C(C)(C)C1CCC1)NC(c1ncoc1-c1ccco1)=O C12(NC(C=C(C)c3ccsc3)=O)CCOC(CNC(=O)C(C)CC(F)F)(C1)C2 C1(NC(C(C)CN(C)C)=O)CCC12CN(C(=O)CSc1cccc(F)c1)C2 Cc1cc(C2CC2)ccc1C(=O)NC1CCC12CN(C(=O)Cc1csc(=N)[nH]1)C2 C(C(=O)NNC(=O)C1CC1C(F)(F)F)OC(C)(C)C.c12cc(ccn1)NC2=O N(C(=NCC1CC1)NCc1cccc(F)n1)C(COC)Cc1ccc(C)cc1 C(=O)(CCCCCC(C)O)NC1CN(C(c2ccc(C)nc2O)=O)CC1O S(=O)(=O)(c1ccc(NCC(O)C(C)(C)C)c(Cl)c1)NC(c1cn(C)cn1)C C1(C(=O)NCC(C2CCC2)NC(C2(CC#C)CCCC2)=O)CCOC1C=C C(C)(C(=O)N(Cc1ccc(C)o1)OC)OC.C1(OC)CO1 c1(C(=O)NC(C(=O)NC(C2CC2(C)C)CC)CC2CCC2)cnc(O)n1CC C(CCCCC(=O)NCCc1cncc(C)n1)NC(C1(CC=C)CCCC1)=O c1(C(N(C2CN(C(=O)CC3(C(F)F)CC3)CC2(C)C)C)=O)ccc2[nH]ccc2n1 c1(C(N(C2CCN(C(C3C(OC)C3)=O)CC2)CC2CC2)=O)cc(Cl)cc(F)c1F c1(OC)cc(F)ccc1NC(=O)CC1CCC(=O)NC1=O C1(C)(CC)CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CN(C)CCOC)C1 CCC(CC(F)(F)F)C(=O)N1CCN(C(c2cnc(C#N)s2)=O)CC1CCOC c1(C(=O)OC)ccnn1CCNC(=O)C1CC1.C1(=O)CCOCCN1C N1(c2cc(CC)nc(C)n2)CCC(NC(c2cccs2)=O)CC(C)(C)C1 O=C(CC1=CCCC1)NC1CCCC(NC(=O)C(O)c2cnc[nH]2)C1 CC(C)CC(C)(C)C(=O)NC(C)Cc1ccc(CNC(C2(C)CC2)=O)cc1 C(=O)(CCCCC(F)(F)F)NC1(C)C2CCC1CC2.N1CCCC(CC)CC1 c1(C(N2C(CN(C(C(C)OCC)=O)C3CC3)CCC2)=O)ccc(O)cc1C Cc1c(C(N2CC(NC(=O)CC34CC(C3)C4)CC2CO)=O)cnn1CCC#N C=CCC(C)(C)CC(=O)NC1CC2CCC1CC2NC(=O)CC1CCC1 CC1CCN(C(=O)CC2C=CCCC2)C(C(=O)NCC23CCCC2CCO3)C1 N1(C(C2N(C(N(CC)CC)=O)CCC2)=O)CC2CC(C1)N(C(=O)C(C)=C(C)C)C2 c1(C(=O)NCCC2N(CC(=O)NCCC)CCSC2)ccc2cccnc2c1 C(N=c1[nH]c(=NCCCC(C)C)[nH]c2c1CCC2)c1cccc(OC)c1 C1(OCC(=O)NCCCN(C(C2(COC)CC(=C)C2)=O)C(C)C)CCC(C)CC1 N1(Cc2c(C)ccs2)CCC(C2(NC(c3cccc(Cl)c3C)=O)CC2)CC1 c1(N2CCCC(C(=O)Nc3c(C)c(Cl)c(Cl)cc3)C2)[nH]cnc2nc(Br)cc1-2 N1(c2nccc(OCCC)n2)CCc2c(NC(C3(CSC)CC3)=O)cccc2C1 C(C(O)CF)NC(=O)NC12CC(C1)C2 CC(=Cn1ccnn1)C(=O)N1CCSCC1CCNC(=O)C(C)n1ccnc1 CC(C)(O)C(F)C(=O)N1CCN(CC(n2cc(NC(=O)ON)nn2)C2CC2)CC1 c1(CC)cc(C(=O)NCC2CC(C(=O)C(O)C(F)(F)F)CN2)cc(O)c1 c1(C(N2CCC(CC(=O)NCc3cc(C)no3)C2)=O)ccc(C)c(C)c1F C1(C2CC2)(C(=O)NC2CC(C)N(C(=O)CC3(C)CC3(F)Cl)C2)CCOCC1 c1(OC)cc(C(N2CCC(NC(C34CC3C4)=O)C(F)C2)=O)ccc1O C1(NC(C=CC(CC)=CC)=O)CCN(C(C2CC(=O)N(C(C)CC)C2)=O)CC1O c1(C(N2C(CCOC)CN(C(C3CCCO3)=O)CC2)=O)ccc2n[nH]cc2c1F c1(NC(=O)NC(CCOC)C)c(F)c(Br)c(F)c(Br)c1F C(C(C)(C)C(=O)NC(C)CCCCNC(C1CCN1S(C)(=O)=O)=O)SC N1(C(C(CCC)N(C)C)=O)CC2(CCN(C(=O)CN3CC4CC4C3)CC2)C1 Cc1ccc(C(=O)NCC2CCN2C(=O)CNc2ccc(C(F)(F)F)cn2)cn1 C(=O)(C(CC)CCCC)NC(CC#C)C(=O)NCCC1CCCC1 C1(OC)CC(NC(=NCCN2CCOCC2)NC2CCOCC2)C12CCC2 Cc1ccnc2nc(C(=O)NCC(O)CNC(c3cc4ccsc4n3C)=O)nn12 N1(C(=O)CCCC2CCC2)CCC2(C1)CN(C(C1CC(=C(F)F)C1)=O)C2 CCCCC(CCCC)NC(=O)CCCCCNC(C1(CF)CC1)=O C1(C(N(C)CC2CCN(C(CC(CC)(C)C)=O)C2)=O)CC2CCCC(C1)C2(F)F c1(C(N2C3CN(C(c4ccnc(F)c4)=O)CC32)=O)cc2cc[nH]c2cc1Cl C(c1ccccc1)(C(F)(F)F)=CC(=O)NC1COC2(C1)CN(C(=O)C(F)F)C2 N1(C(c2nc(C)sc2)=O)CCCCC(N(C)C(C2CC(N3CC(O)C3)C2)=O)C1 CCCCN=C(NCc1cccc(OC(C)C)n1)NC(C)C(C)(C)OC Cc1ccc2c(n1)CCN(C(c1ccc(Br)cc1Cl)C(=O)NC1CCOCC1)C2 c1(CCn2ncc(CN3CCC(N4CC(C)OCC4)CC3)c2)ccc(C#N)cc1 N1(CCc2cn(CC3N(C(c4cc(CC)sc4)=O)CC3)nn2)CC(C)OC(C)C1 C1(NC(c2cn(CC)nc2)=O)CCN(C2CCc3c(F)cc(F)cc32)C1 C1(CNC(c2ccc(OC)nc2)=O)CN(C)CCN1C(C1CC(OC)C1)=O c1(OCCCCCC)ccc(CN(C)C(C2(Cc3ccccc3)CCC2)=O)cn1 S(=O)(=O)(c1[nH]c(=NCC2(OCCO)CCCCC2)ccc1Br)NC(C1CCCO1)C CCC(C)C(O)C(C)C(=O)N(CCC(=O)NC1COCCC1OC)CCCO C(=O)(C(=O)C(C)(C)C)NC1(CNC(C(C)Sc2cnn(C)c2)=O)CCCCC1 C1(NC(=O)OCC)CCN(C(C2CCN(C(C3CC(C)(CC)C3)=O)C2)=O)C1 C(=O)(C1=CCCN(Cc2c[nH]nc2C)C1)NCc1nc(C)sc1 C[S+](C)CCC(O)C(=O)NCC1(O)CCN(C(=O)C(F)C(F)(F)F)CC1 c1(OC(C(=O)N(CC(C)(C)NC(Cc2nc(C)[nH]n2)=O)C)F)ccc(Cl)c(F)c1 CCCCCCCC(=O)NC1CCCN(C(c2scnc2C(C)(C)C)=O)C1 C12(CC(=O)C(=O)CC34CCCC3C4)CCN(N(C3CN(CC)C3)CC)CCC1C2 C1(C(=O)NCc2ccc(CC)o2)(CNC(c2ccns2)=O)CC(C)(C)C1 N1(C(CCNC(N)=O)=O)CCC2(CCCN(C(c3ccc(Cl)nc3)=O)C2)C1 CC(C)(C(=O)NC1CC(O)(CNC(=O)Cn2ccnn2)C1)C1(O)CCC1 c1(C(=O)NC(C)CNC(=O)C(C)(C)c2cc[nH]n2)cccc2c1OC(C)C2 CC1CN(C(C2(O)CCC2)=O)CC1NC(c1ccccc1CC(C)(C)C)=O c1(C(N(C2CCN(C(CC3(C)OCCO3)=O)C2)CC2CC2)=O)cc(F)cc(F)c1 N1(C(CCCC(=O)NC)=O)CCC(NC(=O)CCCOCC)C(F)(F)CC1 N1(C(C(C)OCC(C)C)=O)Cc2n[nH]cc2C1C(=O)NC1CCC(C)C1 C1(C(=O)NCC2CCC(C(=O)NC(C)Cc3cn[nH]c3)O2)CCNC(=O)C1 c1(CCN(C(C(=O)NCC=C)CCc2ccccn2)C)ccc(F)cc1 C1(NC(C(C=C)(C)CC)=O)CCC2(CC1)CN(C(=O)C(C)N1CCCC1)C2 CCC(CC(C)C)C(=O)NCc1ccoc1C(=O)NCCSCC(C)C c1(C(N2CCCC(NC(c3cc(C(=O)OCC)[nH]c3)=O)C2)=O)nc(Cl)ccc1Cl n1(Cc2cccc(OCC)c2)c(SC(F)(F)F)nc2ccccc12 C1(C(NOC(C)CC2CC(C)(O)C2)=O)CCN(C(=O)CCP(C)(C)=O)C(C)(C)C1 c1(C2CCCN(C(C(C#N)C3CNC3)=O)C2)ncc2n1CCCC2 Cc1ncc(C(=O)NCC2(CN(C)C(c3cc(F)cc(Cl)c3)=O)CC2)cc1N N1(C(c2cnc(C(C)C)s2)=O)CCC(C)(NC(=O)C(C)OC2COC2)C1 C12CN(CC3(CCOCC3)C1)C(=O)C1(CC1)NC(=O)C(O)CS2.CN(C)C(N)=O C(=O)(CCCC(=O)NC(C(=O)NCCOCC(F)(F)F)C(C)O)OC N1(C(c2nc(C)n(C(F)F)c2)=O)CCC(C)C(NC(=O)CCN2CCCCC2)C1 c1(NC(C2N(CC)CCCC2)=O)ccc2c(C)nn(C(=O)OC)c2c1 CCCCC(CNC(=O)CC1C(=O)NN=C1C)NC(=O)C(C)=CC(C)(C)C N1(C(c2cc(OC)ncc2-c2cnn3ccccc23)=O)CCC(C)C(F)(F)CC1 N1(C(CC2(OC)COC2)=O)CCOCC1CNC(c1cnc(C)[nH]1)=O CC(C(=O)N(C1CCCC1)CCNC(=O)CCCc1ccccc1)C(F)F C1(C(=O)NCC2CC(NC(C3(C)CCNC3=O)=O)C2)COCCN1C=O c1(C(=O)NCC2CCC(NC(COCCCC(C)C)=O)C2)ccc2n[nH]cc2c1 c1(CCNC2CC(C[Si](C)(C)C)(NC(=O)OC)C2)ccc(O)cc1F c1(C(=O)NC(C=C(C)C)=O)ccc(Cl)nc1C.Cc1nn(C)cc1CO C1(NC(C(c2cncnc2)C)=O)CC(CNC(=O)CN2CC=CC2)CC1O C12(NC(CC)=O)CCCC1CN(C(c1n[nH]cc1Cl)=O)C2 C=CCCCCCCCC(=O)NC1(CNC(=O)C(C)CC(N)=O)CCCC1 CC1=C(C(=O)NCC(O)CNC(C2CCOC2C2CC2)=O)C(C)(C)CCC1 c1(CCC(=O)N(CC(C)NC(c2csc(C(C)(C)C)n2)=O)C)ccccc1 c1(OC)ccc(C(C)C(N2CCCC(n3ccnn3)CC2)=O)cc1OC C1(CCC(=O)NCCCNC(N)=O)CCN(C(=O)CCc2ccc(F)cc2)CC1 N1(C(CC(C(C)C)C)=O)CCOC2(CCN(C(=O)CCN3CCOCC3)CC2)C1 c1(C(N2CCC(C)(CCNC(c3cc(Cl)no3)=O)C2)=O)cc(C2CC2)nnc1O C1(F)(CNC(c2cnn(-c3nccs3)c2)=O)CCN(C(C2COC2)=O)CC1 C(=O)(C1=NN(C)C(=O)CC1)NC12C(CN(C(CCc3c(C)noc3)=O)C1)CCC2 c1(C(=O)NCCc2ncc(C)cn2)n[nH]c2c1CN(C(C1(O)CC(CF)C1)=O)C2 Cc1c(N)ccc(C(=O)NCC2(NC(=O)Cn3ncn(C)c3=O)CCC2)c1F C(=O)(CCC(C)(C)F)N(CC(C)NC(c1ccccc1OCC#N)=O)C CC(C)(CO)C(=O)NCC1CCC(CNC(C2CCOCC2)=O)CC1 C(C)(C(O)C(F)F)NC(CC1N(C(CCSCCCC)=O)CCC1)=O CON(C(=O)c1cccc2c1CCCC2)C1CCS(=O)(=O)C1 C(CCN=c1[nH]c(N2CCN(CC(C)(C)F)CC2)nc2ccc(Cl)cc12)=CC=C C(=O)(C(O)CC(F)(F)F)NCC(C)(C1CCC1)NC(c1c(C)cccn1)=O c1(C(N2CC(O)(CN(C(C(C)n3ccnc3)=O)C)C2)=O)ccnc2[nH]ncc12 c1(NCC2CCCC(SC)C2)ccc(S(=O)(=O)NC(=O)OC(C)(C)C)nc1 CCCCC(CC)C(=O)NCC1C2CCC(C2)N1C(=O)COC1CCOC1 n1(CC)nccc1C(c1nnnn1CC(F)F)NCC(CC1CC1)C1CC1 N1(C(c2c3ccc(C)cc3[nH]c2)=O)CCC(NC(=O)CC2CCCO2)C(C)(C)C1 CN1CCC(C)(C(=O)NCC2CC2CNC(=O)COCC2CC2)C1 CCCCS(=O)(=O)N1CCC(NC(=O)NCC(O)CC(C)C)CC1 CCCC(CC(C)C)C(=O)NC(CC(N1CC2(CCNC(=O)O2)C1)=O)C(C)C CC1(C)C2CCC1(C)C2C(=O)NC1CNCCN1 C(c1ccc([N+](=O)[O-])cc1)=CC(N1CC(O)(CNC(C2CC3CCC2O3)=O)C1)=O Cn1cnc2c1CCCC2C(=O)N1CC(O)(CNC(C2CCCC(F)(F)C2)=O)C1 C(N=c1nc(N2CCCOC(C)(C)C2)c2c([nH]1)CCC2)C1(C)CSCCO1 C1(N(C(CSCC)=O)C)CCCN(C(=O)C(C(C)C)c2ccn(C)n2)CC1 c1(C(N2C(C(=O)NCCCC(C)NC(=O)CCF)CCC2)=O)cccc(F)c1 c1(OC)ccc(C)c(C(=O)N(CCCCN(C(=O)CC23CCC(CC2)C3)C)C)c1 C1(NC(c2cc(C)ns2)=O)CC(Nc2cc(O)ncn2)C12CCC2 c1(C(C)C)ccc(S(=O)(=O)NC2(C)CCOC2)cc1 C1(C(=O)NC2CC(NC(c3ccc(C(F)(F)F)[nH]3)=O)C2)CCC12CCC2 C1(NC(C(COC)O)=O)CC2CCC(C1)N2C(c1ccccc1SC(F)F)=O N1(C(C(=O)NCCSC)c2ccon2)CCCC(c2ccnn2C)CC1 c1(C(=O)Nc2nc(-c3ccnnc3)cs2)c(F)cccc1Br c1(C(N(C2CCN(C(C(C)OC3CCCC3)=O)C2)C)=O)cccc(CO)c1 c1(C(=O)NCCCOCCNC(CSCCC)=O)ccc(-n2ccnc2S)cc1 Cn1c(=O)nc(O)c2ccc(C(=O)NCCNC(C3CSCCS3)=O)nc12 CN1C(=O)CCCC1C(N1CC2C(CC(=O)N3CCC3)C2C1)=O c1(C(=O)NC2CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)c(F)cc(F)cc1Cl C(=O)(CC(C)(C)N(C)C)OCc1nccc(C(=O)NCC(n2ccnn2)C)c1 N1(C(Cc2cccc(C)c2)=O)CCC2C(CCN2C(c2cnn(C)c2C#N)=O)C1 Cc1nc2c(o1)CCCC2CC(=O)NCC1(NC(=O)CCC2CCCO2)CCC1 C(=O)(C1=CCC(C)CC1)N1C(CC)CN(C(=O)C(C2CCOCC2)F)CC1 c1(C(=O)NCC2(F)CC(NC(C3CC3c3ccsc3)=O)C2)cc(F)cc(Cl)c1O C1(C(=O)NCCC(C)N(C)C(C2CSCCS2)=O)CCCC2CCCN12 N1(C(C(C)OCOC)=O)CCC(CNC(=O)C(F)(F)C2CC2)C(C)C1 Cn1ccc2ccc(C(=O)NC3CCCCN(C(C4C=CCC4)=O)C3)cc12 N1(C(CNC(=O)OC)=O)CCC2(CC1)CC(NC(=O)CC1CCCCC13CC3)C2 C1(CNC(C(C=CC)O)=O)CN(c2ncc3ccccc3n2)CCC12CCC2 c1(C(=O)NC2CC(C)N(C(c3cnncc3O)=O)C2)cc2ccccc2o1 C12(CCNC(C3CC(F)(F)C3)=O)CCC1CN(C(C1(CO)CC1)=O)C2 c1(CC(=O)N(CC)CC2CCCN2CC)c(C)noc1Cl.C1(C=O)(CCOC)CC1 Cc1ncccc1C(=O)N(CCNC(=O)CCC1CCCCO1)C1CC1 CC(C)CC(C(=O)N1CC(n2cc(CNC(c3nnc(S)n3C)=O)nn2)C1)C(N)=O c1(C(N2CCC(N(C(C3C4CS(=O)(=O)CC34)=O)CC)C2)=O)csc(S(N)(=O)=O)c1 C1(C(=O)NCC2(COC)CN(C(C(CC)OC)=O)C2)CCCC(C)(C)O1 N1(C(Cc2cc(CC)no2)=O)CCC(C(=O)NCC2(C)CCOC(C)C2)=C(F)C1 CC1CCCN1CC(N1CC(O)(CC(=O)NCCC(=O)OC(C)(C)C)C1)=O N1(C(C2N(C(CN(CCOC)C)=O)CCC2)=O)CCCN(CC2CC2)CC1 C12(NC(C(COC)C)=O)COC(CNC(C3CC(O)CN3C)=O)(C1)C2 C1(C(=O)NCCCC2CCN(C(C(C)c3ccsn3)=O)CC2)CC2(CCC2)CO1 C12(NC(c3ccn(C)n3)=O)CCC(CC1)N(C(c1cc3ncccc3s1)=O)C2 c1(C(=O)NCC(CNC(c2n(CC=C)ccc2)=O)OC)ccc(OC)cc1O C1(C)(CNC(C(CC)OC)=O)CCN(C(c2cn(C(C)C)cn2)=O)CC1 C1(C(C)C)(C(=O)NC2CC(C)(C)C2)CCCN1C(C1C=CCCC1)=O Cc1nc(S(=O)(=O)N2CCC3CN(C)C(C)C23)sc1Br C1(C(=O)NC(c2ccoc2)C)CCC(C)CN1C(c1cccn1C)=O CN1CCC(C(=O)NCCCCCNC(=O)CN2CCCC(N(C)C)C2)CC1=O N1(C(C(CC)(C)OC)=O)CCC(C2(NC(c3cnc(Cl)c(Cl)c3)=O)CC2)CC1 C1(C(=O)Nc2ncc(C)cc2C)CC12CCN(Cc1cc(F)cc(Cl)c1O)CC2 N1(C(c2c(CC)noc2C)=O)CCC(C2CN(Cc3cc(Br)ccc3I)C2)CC1 Cc1[nH]c(C)c(C(=O)NCC(O)CNC(=O)C(O)C(C)C)c1C N1(C(c2c(COC)noc2)=O)CC(C)(C)CC1CNC(C1CN2CCCC1C2)=O c1(C2CC(C(=O)NC(CCOC)CNC(=O)C(C)=C(C)C)C2)ccc(Br)cc1 C(=O)(CC1=NN(c2cccc(F)c2)C(=O)C1)NCC(C1CC1)NC(C(C=C)O)=O c1(C(=O)NC2CC(n3cc(CC(C)(C)CO)nn3)C2)ccc(C2CC2)cc1F CCCCS(=O)(=O)NC(C)C(=O)NCC(CC(C)C)NC(C1(CO)CC1)=O c1(N(CCC)CCNC(c2cncc(F)c2)=O)ccc([N+](=O)[O-])c(SC)c1 c1(CC(=O)NC2CCC(C(=O)OCC)CC2)c(C)nc2ccccn12 C1(NC(C(C=C)C)=O)CN(C(=O)C(C)(C)COCC)CC1CO CCCCCCC(CC)C(=O)N(CC(O)CNC(=O)CNC(=O)CC(F)(F)F)C C12(CNC(C(=O)NCc3scc(C(C)(C)C)n3)=O)CCC(C1)NC2 CCCCCC(C)CC(=O)N1CCC(C(N2CCC(OC3CC3)C2)=O)(CC)C1 Cc1cc(C#N)cc(C)c1-c1cn(CC(=O)NCCCCS(C)=O)nn1 c1(N2CCN(C(c3cccc(F)c3I)C(=O)NCC)CC2)ccc(F)cc1F C1(COC)(NC(=O)Cn2cnc(Br)c2)CCCN(C(=O)C(=O)N(C)C)C1 c1(C(C(=O)NCCC2CC2)N(C)CC)cn2c(F)cccc2n1 c1(CC)ccc(F)c(C(=O)N(C)CC2CC(F)CN2C(c2ccc(N)cc2)=O)c1 c1(C(N2CC3C(CNC(CN(CC)CC)=O)(C3)C2)=O)ccc(C)cc1OC c1(CNC(C=C(C)C(C)C)=O)ccccc1C N(C(=NCC1CC1)NC(c1ccco1)C)CC.N12CCCC1C2=O CCC(C(=O)OC)C(=O)N(CC(N1CCCN(C)CC1)=O)C(C)C c1(C(CC)C)nccc(N2CCCC2C(=O)NC(CC(C)C)c2ccccc2)n1 c1(C(=O)NCC(CC=C)NC(c2ccc(OC)c(F)c2)=O)cc(C)c(CO)cn1 CCC(C(=O)OC)C(=O)NC(C)CC1CCN(C(c2cc(O)ccc2F)=O)CC1 c1(OC)cc(C(F)(F)F)ccc1NC(C1CCCN1Cc1cccnc1)=O Cc1nc(S)sc1CC(=O)NC1CC(C)(NC(=O)CC2COCCOC2)C1 O=C(O)CN1C(=O)COc2ccccc21.C(CO)(CCF)N1CCC1=O N1(C(C2(CC)CC(C)(C)C2)=O)CCN(C(c2cn(C)nc2CC)=O)C(C(C)C)C1 N1(C2C(NC(COCCCOC)=O)COC2)CCN(C(C2(C)CCCC2)=O)CC1 c1(OCCC)ccc(-c2cc(C(=O)OCC3CCC(C)(CC)O3)n(C)c2)cc1F c1(NCC2CCCC(NC(C(C)(C)CF)=O)C2)ncnc2[nH]cnc12 C1(N(C(C=CC(=O)N(C)C)=O)C)CCC(=O)NC1C1CCC1 c1(C(N2CC(CN(C(c3c(CC)n[nH]c3)=O)C)OCC2)=O)cc(Cl)nc(=N)[nH]1 C1(NC(C(CCC)NC(C2CN(C(C)C)C2)=O)=O)CCn2nccc2C1 C12(CNC(C(CCOC)NC(C3ON=C(CC)C3)=O)=O)CCCC1OCC2 CCC(CC(=O)NC1CCCC(C(=O)NC2CC3(COCCO3)C2)C1)CC(C)C CCC(CC)CCCC(=O)NC(CO)C(=O)NC1(C2CCCO2)CC1 N1(C(CNC(CC)=O)=O)CCC2CCN(C(=O)Cc3ccc(F)cn3)C2C1 Cc1cccc(C(=O)NC(Cc2ccco2)C(=O)NC(CCO)C2CC2)c1N Cn1cc(F)c(NC(c2ccn(C3CCC(NCCO)C3)n2)=O)n1 N1(C(CC(C)SC)=O)CCC(C2CCN(C(=O)CC(C)CC(C)C)CC2)C1 Cc1cc(=NC(=O)c2cc(F)ncc2NCc2c(F)cc(Br)cc2F)[nH][nH]1 C1(C(C(=O)NCCOCC)N(CCC(F)(F)F)CC)C2COCC12 c1(C(=O)NCCCCCNC(C2(CF)CCOCC2)=O)cc(Cl)c2c(c1)OCO2 C12(CNC(C(C)CN(C)C(c3cnn(C)n3)=O)=O)CCCC(CO1)C2 c1(C(C)NC(=O)CCC2CCC(NC(=O)C(C)(C)n3cccc3)C2)cccnc1F C(=O)(CC(C)(C)CC(=O)NC1CCN(C(=O)C=CC2CCCC2)C1)OC Cc1cc(C(N2CC=CC2)=O)c(C)n1-c1cc(F)cc(F)c1 C(=O)(CC1=CCN(C(=O)CS(=O)(=O)CC(C)C)CC1)Nc1ncc(C)c(C)n1 C1(NC(c2n(C(CC)C)ncc2)=O)CCCN(Cc2scc(Br)c2C)C1 c1(C(N2CC(O)(CNC(CN(C)CC)=O)C2)=O)cc(CO)ccc1Cl C1(CN(C(C(F)=CCC)=O)C)CCCC(NC(c2cc(C3CCC3)nn2C)=O)C1 c1(CC)occ(C)c1C(N1CCC(CO)(NC(=O)CCc2nc[nH]n2)C1)=O N1(C2C(C(C)C)OCCC2)C(=O)NC(c2ccc(Oc3ccc(Cl)cc3)cc2)C1=O c1(C(N(CCNC(=O)C(C)C2CC2)CC)=O)csc(C(=O)OC)n1 CCC(CC)C(CNC(=O)Nc1cc(C(N)=O)[nH]n1)CO N1(C(C(C)(C)n2cnnn2)=O)CC=C(C(=O)N2CCC(O)CC2)CC1 C(=O)(CC1=CCCCC1)N1CCCC(c2ccccc2)(NC(C2CCC(C)O2)=O)C1 c1(C(=O)NC(C)CCNC(=O)C2=CCCOC2)c(Br)ccc(F)c1N N1(C(c2c(CC)cns2)=O)CCC(C)(C)C(NC(=O)CSc2c(C)n[nH]c2C)C1 CCC(CC)N=C(NCC1(CC#N)COC1)NCC.N1(CC(=O)N)CCCC1 Cc1cn2cc(C(=O)NC3CCN(C(=O)CCn4cccn4)CC3(C)C)sc2n1 C1(CNC(C2CC(C)(C)O2)=O)CCCCN1C(=O)COCc1ccccc1 N1(C(C(C2(C)CC2)NC(c2csc(C)c2C)=O)=O)CCC2CN(C)CC2C1 C(CCC(=O)N1CC(CCCCNC(=O)Cc2ccsc2)C1)SC c1(CC)nc(C(=O)NCC(C2CC2)N(C)C(C2C(C(F)F)C2(C)C)=O)co1 c1(C(=O)NCCOCCC(N2C(C#C)CC2)=O)c[nH]ccc1=O C1(CC(=O)OCC)(NC(=O)C(C)C2CCCC2)CCN(CC(C)SC)CC1 N1(C(C(C=C=C)C)=O)CC2CCC(NC(=O)Cn3c(C)ccc3C)(C2)C1 C(=O)(CC(F)(F)C(F)F)NC(CC)CN(C(C1(C(=O)OC)CC1C)=O)CC N1(C(c2cccc(C)c2)=O)CC(c2cn(-c3ccc(=N)[nH]c3Cl)nn2)CCC1C N1(C(C(NOC)=O)=O)CC2CC(C(N3CC(OCC(C)C)C3)=O)C(C2)C1 c1(SC(C(=O)Nc2cccc(NC(C(F)OC)=O)c2)C)ccn2c1CCCC2 C1(NC(C(CCC)OC)=O)CN(C(=O)COC(F)F)C2CCCCC12 C(C(COC)CC(=O)NCC12CC1CN(C(=O)C(c1ccccc1)=O)C2)OC C(CC(C)C(=O)N1CC(O)CC1C(=O)NCc1snnc1C)=CC CC(C)(C)CC(O)CNC(C1CC(CCNC(=O)C=CCF)C1)=O C12(CNC(c3cnn(C4CCOC4)n3)=O)CC1CN(C(C1CSC1)=O)C2 N1(C(C(C#C)(C)C)=O)CCn2ncc(S(C)(=O)=NC(=O)CC3CCCO3)c2C1 c1(C(N2C(C)C(NC(=O)CNC(c3ccco3)=O)CC2)=O)cccc(F)c1F c1(C(=O)NCC(CO)NC(COc2c(CC)cccc2)=O)cc2cscc2s1 C1(C(=O)NC2C(COC)C2)CC(OC)CN1C(=O)CCN1CCN(C)CC1 CCCC(C(=O)NC(C)CCN(C(=O)C(C)CN(C)C)C)c1ccccc1 c1(CC)cc(NC(C2CC3CC2C2CC32)c2nnnn2C)cc(C(F)(F)F)c1 c1(SCCC(N2C(CNC(c3csnn3)=O)CC(O)C2)=O)ncnc2[nH]cnc12 C(=O)(C(CSC)CC(C)C)NCC1(CC(C(=O)OC)COC)CCCCC1 C1(NC(CN2CCN(C)CC2)=O)CC2CC(NC(=O)Cc3nn(C)cc3Cl)CC12 n1(C(C)(C)C)cnc(C(=O)NCCN(C(C23CCC2C3)=O)CC2CC2)c1 N1(c2ncc(CC)cn2)CCC(NC(c2snnc2C2CC2)=O)C(F)C1 N1(C(C#CC(C)C)=O)CCCC2(C1)C(NC(c1cnn[nH]1)=O)CCN2C C(=O)(CN=S(C)(C)=O)NCC1(NC(CNC(=O)OCC=C)=O)CC1.CO C1(CN(C)C(C2CCCC2CNC(C2(n3cccn3)CC2)=O)=O)CCCC2CC12 c1(NC(CN(CC(C)C)C(=O)Nc2ccco2)=O)ccc(Br)cc1 CC1CC=C(C(=O)N2CCCCC2CCNC(=O)Cn2cc(F)ccc2=O)CC1 C1(C(=O)NCc2occ(C(=O)NCCn3c(C)cnn3)n2)CCCOCC1 C1(CNC(C2(C)CC(F)(F)C2)=O)COCC2(CCN(C(=O)C=CBr)CC2)O1 N1(C(CC(C=C)C)=O)CCCC(CO)(CNC(c2cc(CC)ncn2)=O)C1 c1(C(N(CCNC(c2cnns2)=O)C2CC2)=O)ccc2nccn2c1 N1(C(C(=O)NCCCOCCCNC(C=C(C)Cl)=O)=O)C(C)CCCC1C CCCC(C)(CCC)C(=O)N(CC(C)CNC(=O)Cn1ccc(C(F)(F)F)n1)C Cc1cc(C(=O)NC2CCOCC2NC(C23CCCC2C3)=O)nc(C)n1 c1(C(=O)Nc2c(C)cc(C(=O)OCC)s2)cc(C)c(C)cc1N c1(C(N(C(CN(C(Cc2c(C)con2)=O)C)C)C)=O)ncnc2sccc12 C1(C)(C(=O)NCC(c2ccccc2)C)CCCN1C(=O)CSCC(F)F CC1CN(C(C2(C)CCCS2)=O)CCN1C(=O)CC1OCCC1C c1(CNC(=NCCOC)NCc2cccc(OC(F)F)c2)cc(C)cc(Cl)c1 N1(C(C2C(C)C2)=O)CCC2(CC2)CC1C(N1CCCC(CCO)C1)=O CCCC(C(=O)OC)C(=O)N1CC2(C(N3CC(C)(C)C3C(=O)OC)=O)CCC1C2 C1(NC(c2ccc(NC(N)=O)cc2)=O)CC2CCC1CC2NC(=O)CSC1CC1 N1(C2CCN(C(C3(C(=O)OC)CC(SC(C)(C)C)C3)=O)C2)CCN(C(C)C)CC1 CC1COCCC1C(N1CC(F)CC1CNC(=O)C(F)C1CCCC1)=O N1(C(c2cn(C)nc2O)=O)CC(F)(F)CC1(C)CNC(=O)CCc1ccccn1 C1(NC(=O)Cc2cccs2)CC2CN(C(=O)COCCF)CC2C1 c1(C(=O)NCC(C)NC(C2CN(CC)C(=O)CC2)=O)cc(N)c2ncccc2c1 C12(NC(c3nn(CC)c(C)c3)=O)CCCC1CN(C(c1cc(O)cc(O)n1)=O)C2 c1(NC(C(=O)NC2C=CCN(C(C3(C#C)CCC3)=O)C2)C)cccc(Cl)c1Cl N#Cc1cc(C(=O)NC2CCN(C(=O)CCc3cc(Cl)no3)C2)ccc1[N+](=O)[O-] c1(C(N2CC3C(NC(C(CC)N(C)C)=O)(CC3)C2)=O)ccc(F)c2[nH]ccc12 N1(C(COCCOC)=O)CCC2(CCCN(C(=O)Cc3ccc(C)cc3)C2)C1 C(=O)(CC1=CCN(C(C2OCCC2C(C)C)=O)CC1)NC(C(CCC)C)C N1(C(CC(C)F)=O)CC(NC(=O)C(CC(F)F)NC(=O)OC(C)(C)C)CC(C)C1 c1(C(=O)NCC2C(C)CN(C(=O)CSCC(N)=O)C2)noc2cc(Cl)ccc12 c1(OC)cc(C(=O)NCC=C2CCN(C(C3CCC(=O)N3C)=O)CC2)cc(C)n1 Cc1cc(C(=O)NC2(CC=CC(N3CCCC(CF)C3)=O)CCC2)nn1C C1(NC(c2nc[nH]c2C(F)(F)F)=O)COCCN(C(C2CCCNS2(=O)=O)=O)C1 CCC(F)(CNC(=O)CC(CC1CC1)NC(=O)CCNC(C)=O)CC C#CC1(CCO)COCCN1C(C1CN(C(=O)OC(C)(C)C)C1)=O C#Cc1ccc(C)c(NC(=O)NC2CCC(C(=O)OC(C)C)CC2)c1 C1(CNC(c2nc(C)sc2)=O)CC2CCC1N2C(c1cc2[nH]ccc2s1)=O C1(C#N)(C(=O)NC(c2ccc(F)cc2)(CC)C)CC2CCC1C2 C1(O)(C(C(=O)N(CC(C)C(F)F)C)F)CN(C(=O)OC(C)(C)C)C1 CC(C)C(C)(C(N)=O)NC(=O)NCCC1CCC(C)(C)C1 CC1CN(C(C2CC(C)(C)C2)=O)CC1CCNC(C1CSC1)=O C(=O)(CC(C)CC(C)C)N1CCC(C(=O)NCC)C(O)C1 c1(C(=O)OC)cc(=NC(=O)CC2CCCC2c2ccccc2)[nH][nH]1 CCS(=O)(=O)CCN1CCN(C(=O)NC2CCN(CC(=O)OC)C2=O)CC1 N1(C(c2cc3n(n2)CC(O)CO3)=O)CCOc2ccccc2C1C(F)F C12CCC(CC1)C(=O)NC2.C1(NC(C2(Br)CC2)=O)CC(CF)C1 CC(c1cccc(Cl)c1)=CC(N1CCC(N(C(=O)CN2CCCC2)C)C(C)C1)=O Cc1ccc2c(c1)CN(C(=O)CCN(C(C1(C#N)CC13CCC3)=O)C(C)C)C2 C1C(CO)CNCC=CC(=O)N1.c1(C(=O)OC2CC2)ncoc1C1CCC1 C(C(O)C(F)(F)F)N(C(C)CNC(=O)Cc1csnn1)C c1(CCNC(CCCOCC=C)=O)ccc(CNC(=O)C(F)C2CCC2)cc1 N1(C(COCCC)=O)CCN(C(=O)C(C)CSCc2ccccc2)CC1C c1(C(N2C(c3cn(CC=CC)nn3)CNCC2)=O)nc(C)c2cc(Cl)ccc2n1 C1(NC(c2cc(OCC(F)F)ccn2)=O)C2CN(C(C3CC(O)C3)=O)CC12 C=CC1CC(NC(C2CCCC2OC(C)(C)C)=O)C1 C12(C(=O)NCC(CC)N(C)C)CC(C)(CN1C(=O)C(C)SC)C2 C(=O)(C(C)CCC(C)(C)C)NCC(c1nc[nH]n1)C.C12CCC(C1)NC(=O)CC2 N1(C(C2(COC)CCCO2)=O)C2CCC(C2)C1CNC(C1C(C)(C)C1(C)C)=O C(=O)(CCCC(=O)N(C1CCN(C(=O)CN2CCC(C)C2)C1)C)N(C)C Cc1oc(C#N)cc1C(=O)NCc1nocc1C(=O)NCC12CCCC1C2 C=CC1(C(=O)NC2CC(CCNC(c3cc(CC(C)C)[nH]n3)=O)C2)CCCC1 C1(CNC(c2ccc(-c3ccc(Cl)s3)s2)=O)CCCC1NC(C1(O)CCC1)=O C1(NC(c2cc3ncccc3[nH]2)=O)CC12CCC(NC(C1(Cl)CC1)=O)CC2 c1(OC)ccc(OC)c(OC)c1-c1noc(CC2(C)NC(=O)NC2=O)n1 C1(C(=O)NCC(C)NC(c2ccccc2C2CCOC2)=O)C2CCC1CC2 CCC(C(=O)NCC(CCOC)NC(=O)Cc1c(C)nc(O)nc1O)C(F)(F)F N1(C(C2C(C)(C)OCC2)=O)CCN(C(c2nn[nH]c2Cl)=O)C(CC(F)(F)F)C1 CC(C)(C)C(CCc1ccc(F)cc1)NCc1ccc([N+](=O)[O-])o1 C(=O)(C(O)C(F)(F)F)N1CCC(C(C)NC(=O)Cc2cnn(C(F)F)c2)CC1 C1(CNC(c2cnsn2)=O)CC12CCN(C(c1n[nH]c3c1CSCC3)=O)CC2 C(=O)(CS(=O)(=O)CCO)NC1CCCC(NC(c2cccc(C)c2)=O)CC1 c1(CC(=O)NC(C)CCNC(c2ncn(C3CCCCC3)n2)=O)cccc(Cl)n1 N12CCN(C(=O)C1)CC2=O.c1(OC)cc(N(C2CNCC2O)C)[nH]n1 N1(C(C2C(C=C)OCC2)=O)CCC=C(C(=O)N2CCOC(C3(C)CC3)C2)C1 Cc1ccc(C(=O)CCN(c2ccccn2)Cc2ccccc2)cc1 N1(C(C(C)NC(COC)=O)=O)CCN(C(c2cscn2)=O)CC(C)(F)C1 N1(C(CCCC(CC)CC)=O)CCCC2C1CCCCN2C(=O)C=CS(C)=O C=C1Cn2c(C(=O)NC3CC(NC(C4(OC)CCSC4)=O)C3)nnc2S1 C1(OC)CC(C(N2C(C(=O)OC)CC2C)=O)N(C(c2sc(CO)nc2C)=O)C1 C1(C(=O)NC(C2CN(C(c3cc4ccsc4s3)=O)CCO2)C)CCCCN1N=O C1(NC(C2CC(=O)N2)=O)CN(C(c2cc3occc3s2)=O)C2(CCOCC2)C1 C1(NC(C2(OCC)CCC2)=O)CCCC(NC(=O)C(CF)=CC2CC2)CC1 Cc1cc(Cl)cc(C(N2CCCC(N(C(=O)CCC(C)(C)F)C)C2)=O)c1N(C)C CC(C)C(F)(CNC(C1(CO)CCCO1)=O)C(=O)N1CCCCC(CO)C1 C1(NC(COCC(C)C)=O)(CO)CCCN(C(c2cncc(F)c2)=O)C1 S(=O)(=O)(c1ccc(F)cc1)NCC(=O)NC1CCOCC1NC(=O)CC(=O)NCC1CC1 C1(CNC(CNC(CC(C)C)=O)=O)CC12CCN(C(=O)CNS(=O)(=O)C1CC1)CC2 c1(CC)cc(C(N2CCCCC2CNC(C2CC2COC)=O)=O)ccc1O Cc1ncc(C(N2CC(C(=O)NCc3cccnc3O)C(C(C)C)C2)=O)c(C)n1 CC1(C#CC(=O)NC2CC3(C2)CC3C(=O)NC2CC3CCCC3C2)COC1 c1(NC(C(C)N2CCCC2)=O)ccccc1C(=O)NCCN1C(=O)CNC1=O N1(C(C2N(S(CCCC)(=O)=O)CCCC2)=O)CCN(C(c2cn[nH]c2)=O)C2CC12 c1(CC)ccc(F)cc1NC(=O)C(C(C)C)NC(=O)Cc1sccc1C C(=O)(C(C(C)C)C(C)C)N1CCC(N(C(c2ncc(C)c(Br)c2)=O)C)C1 CN1CCn2ncc(C(=O)NC3CN(C(=O)C=Cc4cccs4)CC3O)c21 CC12CCCN1C2=O.c1(CNC(=O)C(c2ccccn2)O)ccccc1 C(=O)(C1=CCOCC1)N(C1CCN(C(C(C)CC2CCCCC2)=O)C1)CCO c1(C(N(CC(C)N(C(Cc2c(C)ncs2)=O)C)C)=O)cc(OC(F)F)cc(F)c1 N1(C(Cn2cnc(C#N)n2)=O)CCCC2CN(C(C3CCCC3(F)F)=O)CC12 C1(NC(CCSCCNC(CCC2CCC(=O)C2)=O)=O)CC2C(O)C(O)CC12 N1(C(c2cc(C)c(F)cn2)=O)C2CCC1CC(C(=O)N(C1CCCNC1=O)C)C2 C(CCC(=O)NCC(C)NC(C1CC1c1cnn(C(C)C)c1)=O)N(C(=O)OC)C n1(CC(=O)NC2CCC(F)(CNC(C3CCOC3)=O)C2)nc(Cl)ccc1=O N1(C(C2NC(=O)OC2)=O)CC2CC(NC(c3ccnn3C3CC3)=O)C1C2 N1(CCn2cc(CC(=O)OC)nn2)CCN(C(=O)C(C)(C)C)CC1 C1(C(=O)NCCCOCCNC(C2CC(n3cnnc3)C2)=O)CC1[N+](=O)[O-] C(=O)(CC1=Cc2ccccc2C1)NCC1N(C)CCN(C(c2cc(C)no2)=O)C1 N12CCC(C3CC3)C1C(=O)NC(CC1CC1)C21CC1.c1(OC)ncc(C=O)cn1 CCC(C(=O)N1CCC(CC2CCN(C(C3(O)COC3)=O)CC2)CC1)C(C)C C1(C(N(C2CCN(C(c3cnn(CC(F)F)c3)=O)CC2)C)=O)CCC2(CC1)N=N2 C1(C(C(=O)N(CC(C)NC(c2c(COC)scc2)=O)C)O)CCCCCC1 O=S(=O)(c1ccc(NCC2COCO2)cc1Br)NCc1cc(F)c(Cl)cc1Cl C(=O)(C(C)(CNC(=O)C(=O)NC1CCOC1)CC)Nc1ccc(C(=O)OC)cc1 C12(C(=O)NCCN(C(=O)CCCCCSC)CCOCC)CCC(CC1)C2(C)C N1(C(CC(C=C)C)=O)CCc2sc(CNC(C3CC4(CCC4)CCO3)=O)nc2C1 C1(CCC)C(=O)NCCN1C(=O)N(CCCN(C)Cc1ccc(C)cc1)C C1(NC(C(CC)(C)C(N)=O)=O)CCC2(CC1)CCN(C(=O)C1=CCCSC1)CC2 C(CCCCCC(=O)NC1(c2cccs2)CC1)NC(C(C=C)OC)=O N1(C(c2n(COC)ncc2)=O)CCC(C(=O)NC2CCCCC2)C1(C)C N1(C(c2ccn(C)c2)=O)CC2CCN(C(=O)C3=NOC(CC4(O)COC4)C3)C2C1 C(C)(CNC(c1ccnn1C)=O)(CC(C)C)NC(C(C)OCCC(C)C)=O c1(C(=O)NCC(C)NC(C=NOC)=O)cc([N+](=O)[O-])ccc1Nc1ccccc1 C1(CNC(C2CC(=C)C2)=O)CN(C(=O)CCc2ccc(C(F)(F)F)cc2)CCO1 C1(C(N2CC(NC(c3cn(C)c(=O)cn3)=O)CC2(C)C)=O)CCn2cnnc2C1 C=CCC(CC)C(=O)NC1CCC(C(=O)Nc2cnn(C)c2C(C)C)CC1 C1(NC(C2C(C#C)C2(C)C)=O)COCCN(C(=O)CSc2ccc(F)cc2)C1 C=C=CCCC(=O)NC(C)(C)CC=CC(=O)NCC1CCCC1CF C12(CNC(c3c(C)cco3)=O)CCC1CN(C(=O)CCC1(C)CC1)C2 c1(C(=O)NC(CNC(C(CCCCC)O)=O)(C)CO)[nH]nc2c1CCCC2(C)C N1(C(C2CN(C)C(=O)N2)=O)CCN(C(c2scnc2Cl)=O)C2COCC12 c1(OC)nc(C)ccc1C(N1CC(NC(=O)CCCNC(N)=O)C(O)C1)=O CN1C(=O)CCC1C(=O)NCC(CO)NC(c1cn(C2CCOCC2)cn1)=O C(=O)(C=C1SCC(=O)N1C)N1C2C(NC(CC(=O)NCC#C)=O)(CCC2)CC1 Cc1nc2cc(NC(N3CCC(Cc4cc(Br)c(C#N)s4)C3)=O)ccc2s1 c1(C(=O)NC2(CNC(c3ccc(F)s3)=O)CC2)c[nH]c2ccc(F)cc12 CCCCC(C)(F)C(=O)NC(C1CCCN1C(=O)CSCC(N)=O)C N1(C(C(CC=C)NC(=O)CC#N)=O)CCN2CC(C)CC2C1 CCC(O)C(C)C(=O)NCC1CCN(C(=O)C=C(Cl)Cl)C1(C)C N1(C(c2c(CC)n[nH]c2)=O)CCC(F)(CNC(C2(C3CCCO3)CCC2)=O)CC1 c1(C2N(C(C3(O)CCCCCC3)=O)CCC2)ccc(NN2C(=O)CCC2=O)cc1 Cc1csc(NC(C)C(N2CCC(CCC(=O)NCCc3csc(C)n3)C2)=O)n1 C1(OC)CN(C(c2cc(C)on2)=O)CC1NC(c1cc(F)cs1)=O C1(NC(C2C(c3n(C)c(S)nn3)CCCC2)=O)CCN(C(=O)OC(C)(C)C)C1(C)C C(C(N=[N+]=[N-])C(=O)NCCCC(=O)NCc1cc(F)ccc1O)OCC N1(C(CC)=O)CCC2C1CCCN2C(c1cnccn1)=O C1(CNC(c2ccc(SC)o2)=O)CN(C(c2cscc2F)=O)CCC1(C)C c1(C(=O)NC2CN(Cc3c(Cl)ccnc3Cl)CC2O)cc2cccnn2c1 c12cc(c3cn[nH]c3c1)NC(=O)Cc1ccc-2cc1.c1(CN)ccc(Br)s1.N#CC N1(C(C2CN(C)C2)=O)CCC(NC(=O)C=CC2CCC2)C(C(N)=O)C1 C1(CCNC(=O)Cc2cc[nH]n2)CN(C(c2nc(Cl)c(Cl)s2)=O)CCO1 c1(C(N2CCCN(C(C(CCOC)C)=O)CC2)=O)n[nH]c2cccnc12 N1(C(c2cncc(NC)c2)=O)CC23CCCC2(C1)CN(C(C1CC1F)=O)C3 Cc1ccc(C)c(CNc2nccc(N3CCCC(F)C3)n2)n1 C1(C(N(CCCCCC)C)=O)CN(C(C2CCCCN2C)=O)CCO1 C1(CNC(C(=O)NC(C)C)=O)(NC(c2cc(C(N)=O)co2)=O)CCCCCC1 N1(C(c2c(C)csn2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 C1(C)(C(=O)NCCCOCC=C)CN(C(=O)CC2CC2C2CC2)CC1C c1(OC)cc(C(N2CCN(C(C3CC(=O)CC3C)=O)CC2)=O)ccc1I Cc1ccc(F)cc1COC(C1CN(C(=O)OC(C)(C)C)CCC1F)=O N1(C(CCSC)=O)Cc2ccccc2C(NC(C2(F)CCOC2)=O)C1 N1(C(C2C(OC)(OC)CC2)=O)CCCC(C(=O)Nc2ccc(NCCO)cc2)C1 c1(C(C)C)nc(N(C)CCNC(=O)N(C)C)cc(N2CCC(O)C2)n1 c1(C(N2CC3C(CNC(C4(COC)COC4)=O)C3C2)=O)cncc(C(F)F)c1 N1(C(C2C(C)C2c2ccccc2)=O)CC2CC2(CNC(=O)CSC2CC2)C1 c1(C(C)(C)C)n[nH]c(=NC2CC3CC(C2)N(C(=O)CC2=CCCCC2)C3)o1 CN1C(=O)OCC12CN(C(=O)C(CCN(C)C)NC(C1CC13CCOCC3)=O)C2 N1(C(CC(C)C2CC2)=O)CCC(NC(c2nn(C(F)F)cc2Cl)=O)CC(C)(C)C1 Cc1cncc(C(=O)NC(C)CCCNC(c2cc[nH]c2C2CCCC2)=O)n1 C1(NC(Cn2ccc(C)n2)=O)CC2CCC(C1)N2C(=O)Cc1csnn1 c1(C(N(CCNC(c2cscc2SC)=O)CC)=O)ccc(N)c(F)c1 Cc1ccc(C(C)CC(=O)OCc2cccnc2C)cc1 N1(C(C(CC)NC(N)=O)=O)CCC(C)(CCNC(c2ccc(OC)cc2)=O)CC1 C1(OC)(CNC(C2CC2(C)C)=O)CCN(C(c2cscc2-c2ccccc2)=O)C1 C(=O)(CC(C)(C)C(F)F)N1CCN(C(C2C(=C)C2)=O)CC1c1nccn1C c1(OC(C)C)cnc(C(=O)NCC2CCC(NC(C3CC(C)(F)C3)=O)C2)cn1 N1(C(C=CCN(CC#C)C)=O)CC2CC(C)N(C(c3cc(C)n(C)c3)=O)C2C1 C1(CNC(C(COC)OC)=O)CC2(CCN(C(c3csc(C)c3N)=O)CC2)CO1 C1(C(=O)NCc2ccnc(OC)n2)CN(C(=O)CC2OCCCO2)CCN1C c1(C(C(=O)NC(CC)C)N(C)Cc2ccc(F)cn2)ccc(C)cn1 N1(C(COCC(=C)C)=O)CC(F)(F)CC1CNC(c1cc2[nH]ccc2s1)=O CC1(C)CCC(C(=O)NC(C)(CNC(=O)COc2ccon2)C2CC2)C1 C(=O)(CC(CNC(C1(C)CC1(F)F)=O)N(C)C)NCCc1onc(C)n1 c1(C(N(CCOC)CCNC(c2c[nH]nc2F)=O)=O)cc(C)cc(Cl)c1 Cc1cc(C)c(C(=O)NC(C(=O)N(C2CC2(C)C)C)c2cccs2)cn1 C1(C(=O)NCCC(=C)C)CC(NC(=O)CCc2cnn[nH]2)CCO1 Cc1c(CNC2CN(c3cccc(Cl)c3)C2=O)c(C#N)c2n1CCC2 C1(C(=O)NCC(CC=C)NC(C2CC(OCC)C2)=O)(CF)CC(F)(F)C1 c1(N2CC3CC(NC(c4ccoc4)=O)C3C2)ncnc2sc(C(F)(F)F)nc12 CC1(C(=O)NCCNC(C2CC(c3cccc(F)c3)(F)C2)=O)CCCOC1 n1(C(=O)NCC2CC(OC)CN2C(c2sc(CO)nc2C)=O)ccc([N+](=O)[O-])n1 C(=O)(CCC(CC)CC)NC(CSCC)C(=O)N(C1(C)CCCC1)C C1(CC(C)C)CCN(C(C2CCC(CNC(c3csc(CO)c3)=O)C2)=O)C1 c1(OC)cc(I)ccc1C(N1C2CN(c3cccn4cncc34)CC12)=O c1(C(c2nnnn2CC)NC(COCC)C)ccccc1-c1ccccc1 Cc1cccc(F)c1C(=O)N(CCC(C)NC(c1cnn(C)c1Cl)=O)C N1(C(c2ccsc2Br)=O)CCOC(CNC(C2(n3cccn3)CC2)=O)C1 Cc1nc(C(=O)N(c2ccc(I)cc2)n2cncn2)ccc1-c1ccccc1 c1(-c2c(C)c(F)ccc2)ccc2c(c1)CCN(C(c1ccc(Cl)cc1I)=O)C2 c1(C(=O)NCC2N(C(Cc3c(C)ocn3)=O)CCOC2)cnc2c(Cl)cccn12 CC#CCCCC(=O)N1CCC(C(=O)N(C2CCN(CC)C2)C)O1 C(=O)(C(N=[N+]=[N-])C(C)C)N(C(C(=O)NC(C(=O)OC)CO)CC(C)C)C CC(CC(=O)NC12CC(CNC(C3(F)CCOC3)=O)(C1)C2)C(F)F C1(N(C)C(C2CSCCS2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C C(=O)(CC(C(C)OC)NC(=O)C(N1CCCCC1)C)NC(c1cscn1)CC c1(C(=O)Nc2ncc(CC(C)(C)O)s2)nc2cc(F)ccc2s1 CCC(C)CC(=O)n1cc(C2(F)CN(C(=O)C=CC(C)C)C2)nn1 CC(C)C(CC1CCCCC1)C(=O)N1CC2CC1C2NC(=O)Cn1ncnn1 C1(C(=O)NC(CNC(c2cc(-c3ccc(C)s3)[nH]n2)=O)(C)C)CC2C(C1)C2(C)C c1(Cn2cc(C3N(C(c4sc(SC)c(Br)c4)=O)CCC3)nn2)cc(Cl)ccc1Cl C=C1CCC(C(=O)NC2CC(NC(c3cc(C)[nH]n3)=O)C2)CC1 Cc1cc(N2CCCC(CN(C)C(c3sc(C)nc3C)=O)C2)nc(C)n1 c1(CC(=O)N(C)CC2N(C(CN(C)S(N)(=O)=O)=O)CCCC2)ccc(F)c(F)c1 N1(C(c2ccc(C#C)cn2)=O)CC2CC1CN(C(C1CCCOCC1)=O)C2 C1(C(C)NC(=O)CN2CCC(CO)C2)CCCN(C(=O)Cn2ccnc2)C1 N1(C(C(CC)CC2CCCC2)=O)CCN(C(=O)C(C)(C)CF)CC1CCOC C1(C(C)C)CCN(C(C2CCC(C3CC3)N2C(c2cnc(=N)[nH]c2)=O)=O)CC1 N1(C(COC)=O)CCN(C2CCCN(C(=O)Cc3ccco3)C2)C(=O)C1 c1(C(N(CCNC(=O)CC(C)CC)CC)=O)cc(F)c(F)cc1O C(=O)(C(C(C)(C)C)NC(=O)Cc1ccon1)NC(c1ncn[nH]1)C c1(CNC2C(CC(C)C)CCC2)cnc2c(C(N)=O)cnn2c1 CC(C)(CCCC1(C)C(C(C(=O)OCC)C#N)C1)NC(=O)CCc1ncc(F)cn1 C1(C(N2C(C)CC(NC(CC=C)=O)C2)=O)CC2CC1C1CC21 Cc1ccc2oc(N3CCC(NC(=O)CC4CC4(Cl)Cl)CC3C)nc2c1 Cc1cc(F)ncc1C(N1CCC1CNC(=O)C(CO)NC(c1ccco1)=O)=O C1(CN(C(CCNC(=O)OCC)=O)C)CC(C(=O)N(C)CC2CC2)CO1 N(C(=NCc1cccc(CC)c1)NCc1ccn(C)n1)C(C=C)C C1(CNC(C2(CC(C)C)CCC2)=O)CCC(NC(=O)Cc2c(Cl)cnn2C)CC1 N1(C(C2(C#N)CCCO2)=O)CC2(CCC2)CC1C(=O)NCCN1CCCNC1=O N1(C(C(CCC)CC)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC(O)C1 C1(NC(C(CC=C)CC(C)C)=O)CC(N=c2[nH]c(C3CC3)nc(Cl)c2C)C1(C)C N1(C(CC2(OC)CN(C(C(CC)n3ccnc3)=O)C2)=O)CCOCC1C1CCC1 C1(C(=O)NCc2ccc(C(=O)NC3(CC(N)=O)CCCC3)o2)CC(=O)CCO1 C(=O)(C1=NOC2(CCOC2)C1)NC(CCNC(c1cnc(C)o1)=O)C C1(CC(=O)NOCC2CCOC2)CC2(C1)CN(C(=O)Cc1ccc(Cl)cn1)C2 c1(C(=O)NCC2CN(C(C(C)n3cccn3)=O)C(C)(C)C2)ncn2c1COCC2 C1(C(N(CC(C)O)CCNC(c2cc(CC)ncn2)=O)=O)CC(C)(C)OC1(C)C C1(CN=C(N(C)Cc2ccc(Cl)o2)NC2CC2)CC2COCC(C1)C2(F)F n1(-c2ccn(CC)n2)nc(C(C2CC2)OC(C)(C)C)nc1-c1ccsc1Cl CC1(C)CC(C)(C(=O)NCC2CC(C(=O)NCCCCC3CC3)C2)C1 N1(C(CCOC(CC(C)C)C)=O)CCC(O)(CCNC(=O)CSc2cccs2)C1 C1(C2(O)CN(C(=O)C(C)(C)CSCC)C2)(CNC(CC(=C)C)=O)CC1 c1(C(C)C)nc2ccccc2n1CC(=O)NCC1CN(C(=O)C(N)=O)CCC1C C1(CC(=O)N(CCCNC(CCNC(=O)CO)=O)CCO)CCCCC1O c1(C(=O)NC(C(C)NC(Cc2scc(CC)n2)=O)C)cc(C(F)F)nn1C c1(OC)ccc2c(c1)CCC2C(=O)N1CCC(C)(NC(c2ccsc2C)=O)CC1 C12(NC(C(C3CCC3)OC)=O)CCCC1N(C(C1(F)CCC(=O)CC1)=O)CC2 CCC(C)CC(C)N(C(=O)CC1CN(C(=O)CSC)CCO1)C1CC1 C1(C(N(CCN(C(C)C)C(c2cnccc2Br)=O)C)=O)CCC12CCC2 CCCCCCC(C)(CCC)C(=O)NCC1CCN(Cc2ccccc2)C1=O CC1CCC(NC(C2(c3cccs3)CC2)=O)CN1c1cc(C(C)(C)C)nc(Cl)n1 C1(NC(C(C(COCC)C)C)=O)CCN(C(=O)CN(C)C(=O)OC)CC12CCC2 N1(C(=O)CCc2cccc(NCc3nn[nH]n3)c2)CCOCC1C1CCOCC1 CCCC(C)CCCC(=O)NCCC1(CNC(=O)CCCCCOC)CCCC1 C1(NC(C2(CCC)CCC2)=O)CCN(C(=O)CCNC(=O)C=CCl)CCC1CO c1(C(N(C2CCN(C(C3CCOCC3)=O)C2)CC)=O)ccc(C)nn1 C1(NC(C(CC)NC(N)=O)=O)CCC(CNC(=O)C2CC2)CC1.C1C(=O)N1 N1(C(C2C(C(N)=O)C2)=O)CC2CCC1CN2C(=O)Cn1ccc(C(F)F)n1 C1(NC(C=NOC)=O)CCN(C(c2cc(C)nc(C)c2)=O)CC(C)(C)C1 C(=O)(CC(CC)C(C)C)N(CCC(C)NC(C1(COC)CCCC1)=O)C N1(C(C2CCCN(C(C(C(=O)OCC)OC)=O)C2)=O)CC2CCC1CC2 C1(CNc2cc(C)ncn2)CCCN2CCCC12.c12ccc(cc1F)[nH]2 c1(NCCc2c(C)nccc2)nccc(=NC2CSC(C)C2)[nH]1 c1(SCC)cnc(O)c(C(=O)NC2CCCCC2NC(c2snnc2CC)=O)c1 c1(NC(=O)NC)ccc(C(=O)OO)c(F)c1.C(C)(C(C)(C)C)=CC(=O)NC(C)=O NC(=O)C#CC(=O)N1CCC(C2OCCC2NC(c2cnc(Cl)s2)=O)CC1 C1(C)(C(=O)NCC(CCOC)(C)O)CCCN(C(=O)C=CC(F)F)C1 c1(C2C(NCC(COC(=O)OC(C)(C)C)(C)C)C2)ccc(F)cc1Cl c1(C(=O)NCC2COCC2NC(c2cnc[nH]2)=O)cncc(CO)c1 CCC(C)CC(=O)NC1CC(CNC(c2occc2COC)=O)CC1O N1(C(C(CC)CC)=O)CC(NC(=O)C(C)(C)CSC)CC12CCCOC2 c1(NCC2C(CNC(C3=C(C)OCC3)=O)C2(F)F)cc2nnc(C(C)C)n2cn1 c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)C#N)cnc2sc(C)cn12 N1(C(COCCOC)=O)CCC(NC2CCN(c3nc(C(=O)OC)ns3)C2)CC1 Cc1ccc2[nH]cc(C(=O)CNC(=O)CC3CCCCNCC3)c2c1 CC1(C)Cc2[nH]nc(C(=O)NCCC3CCCCN3C(=O)C3=C(Cl)CC3)c2OC1 N1(C(C(CCC)NC(N)=O)=O)CCOC(C(=O)N(CCC2CCC2)C(C)C)CC1 C#Cc1ccc(C(N2CCC(CNC(C3CN(C)CCO3)=O)C2(C)C)=O)c(C)c1 C1(CC(=O)N(C(CNC(c2ccc(C)nc2)=O)C)C)CCCCC1(F)F Cc1cc(C(=O)NC2CC2NC(c2csc(C(C)(C)C)c2)=O)nc(O)n1 C1(CC(=O)O)CCN(CC2CN(CC3CC3)C(=O)O2)CC1(F)F c1(C(=O)NCC2(O)CCCC2)ncn2cc(-c3cccc(O)n3)sc12 Cc1cc2c(C(=O)NC(C)CC(C)NC(c3c(C)ccn3C)=O)ccc(C)c2[nH]1 C1(C(N2CCC(NC(CCN(S(C)(=O)=O)C)=O)C2)=O)CC(S(C)(=O)=O)C1 N1(CC(=O)NC2C(CNC(CCCC)=O)C2)CCN(C(C)=O)CC1 N1(C(C2(C#N)CCC2)=O)CCC2CCCN(C(c3ccccc3O)=O)C2C1 c1(C(=O)NCC2N(C(c3c(C)scn3)=O)CCC2)cc(F)c(F)c(C#N)c1F c1(CC(=O)NCCCNC(C23COC(CO)(C2)C3)=O)ccc2c(c1)OCCO2 C1(C(N2CCCCC2C2CNC(=O)C2)=O)CC2(CCC2N)C1 C(CC(C(C)(C)C)NC(=O)Cc1cnco1)N(C(c1c(C)snc1)=O)C c1(C(=O)NCC=CCNC(=O)CCSC(F)(F)F)ccc(Cl)c(F)c1O N1(C(C2CN(C(C3(C)CC(C)C3)=O)CC2C(C)C)=O)CCCNC(=O)CC1 C1(NC(Cn2c(C(C)C)ncc2)=O)CC12CC(NC(c1ccc(F)cc1)=O)C2 c1(C(C)OC(c2nscc2Br)=O)ccc(-n2ccnn2)cc1 C1(CC(=O)N(C2CCNCC2)C)CN(C(=O)CSc2ccccn2)CCS1 C(C)(CCC(=O)N1CCC(C)(F)C1)NC(CC(C)=C(C)C)=O Cc1ccnc(-n2cc(C(=O)NC3CCN(C(c4cc(C5CC5)on4)=O)C3)cn2)c1 n1(CC)nc(C)c(C(=O)NCC2(NC(C3C4CCCC34)=O)CC2)c1Cl C12(CNC(NCC(C=C)(C)C)=NCCc3ccccn3)CCC(COC)(CO1)C2 N1(C(C(C)=CC)=O)CCN(C(=O)C(C(C)C)c2cccc(C(F)(F)F)c2)C(C)C1 S(=O)(=O)(c1cccc(C(=O)Nc2ccccc2)c1)NCC1CC12CC2 CCCCCC(C)CC(=O)N1CCSCC1CCNC(c1ncc(O)cn1)=O C1(C(=O)NC2(C)CCCC2)C2CC2CN1C(c1ncc(F)cn1)=O N1(C(C(C(C)(C)C)OC)=O)CCN(C(=O)CCC(C)(C)C)CC12CC2 c1(C(=O)NC2CC2C(=O)NCCOCCO)ccc(CCO)cc1.CO c1(C(=O)NC(C2CCN(C(C3CNC(=O)N3)=O)CC2)C)ccnc2c1ncn2C C#CCC(C)(C(=O)NC(c1nnc(O)n1C)C)NC(=O)C(O)C(C)(C)C O(NC(=O)C(CC1CCCC1)C(C)C)Cc1cn(-c2cccc(C)n2)nn1 C1(C(=O)NCC(CNC(c2cc(CCC)n(C)n2)=O)OC)CS(=O)(=O)CC(=O)N1 C(=O)(C(Cc1cc[nH]n1)NC(c1cnsn1)=O)NCC(C)F N#Cc1c[nH]c(C(=O)NC2(CN(C(=O)CCCn3ccnc3)CC)CCCCC2)c1 N1(C(C=C2CCC(C)CC2)=O)CCN(C(C2CCCCCN2C)=O)CC1C c1(OCC(C)NC(=O)NCC(n2nccn2)Sc2ccccc2)cccnc1 c1(C(=O)NC2C(n3cc(CC(=O)NC)nn3)CCC2)cc(F)c(Cl)c(OC)c1Cl c1(NCC(CC)(CC)NC(=O)CS(=O)(=O)NC(C)C)nc(Cl)nc2c1cnn2C N1(C(c2cc3ncccc3[nH]2)=O)CCC2CCC(NC(C34CCC3C4)=O)C1C2 Cc1ccc(F)c(CNC2CCCCC2NCC(N)=O)c1 N1(C(C2C(CC)CN(C(=O)CC3CCC3)C2)=O)CCCCCC1C(C)C CCCC(CC(C)C)C(=O)N1CCCC12CCN(C(=O)CNS(=O)(=O)CC)C2 C1(C(=O)NCCCNC(c2c[nH]nc2Cc2ccccc2)=O)CC2C=CC1C2 N1(C(CCCCNC(COCC(=O)OC)=O)=O)CCCC(C)(C#N)C1 c1(NCc2cccc(NC(N(C)C)=O)c2)cccc2c(F)ccnc12 CCS(=O)(=O)CC(=O)NCC(C)NC(c1cccnc1NC1CCN(C)C1)=O c1(C(=O)NC(CNC(C(CCCC)(C)F)=O)C)[nH]c2c(c1C)CCCC2 c1(C(N2CCCC(NC(C3C(OC)CCCCC3)=O)C2)=O)cc(C#N)cc(C)n1 C(=O)(C#CC(C)(C)CNC(C1CC=C(C)CC1)=O)NCCSCC#C c1(CC(=O)N(C)CCNC(c2cc(C3CC3)on2)=O)ccc(S(=O)C2CC2)cc1 c1(OC)ccc(CNCCC2CCCCO2)cc1 C12(NC(CNC(=O)NC)=O)CCOCC1CN(C(=O)CCC=CBr)C2 O=S(=O)(c1[nH]c(=NC2CC(CF)C2)ccc1Br)NC1CCOCC1O Cc1c(NC(C2(C(C)C)CCCN(C(=O)OC(C)(C)C)C2)=O)c(Br)nn1C N1(C(C#CC)=O)CCn2nc(CNC(C3CC(S(C)(=O)=O)C3)=O)cc2C1 C1(C(=O)NC2C(C)(C)CC2NC(C2CN(CC(F)F)C2)=O)CC12CCOCC2 CC1(C)CCCC(CS(=O)(=O)NCC2CCCCN2Cc2noc(C3CC3)n2)C1 c1(C(C)C)nnc(C2CC2C(F)(F)F)n1C1CCC1.C12CC(C1)NC2 N1(C(C=CCN(C)CC)=O)CCCC(O)(CNC(C2CC2(Cl)Cl)=O)CC1 N1(C(c2ccc(C)cc2C2CC2)=O)CCC2CN(C(=O)C(C)(C)OC(F)F)CC12 C1(S(N)(=O)=O)(C(=O)NC(C2CN(C(=O)CC(C3CC3)C3CC3)CCO2)C)CCC1 n1(CC(=O)NC2(CNC(=O)CC3CCC3)CCCCC2)ccc([N+](=O)[O-])n1 c1(SCCC)ccc(C(=O)NC2CC2NC(=O)COC(C)C)cc1.CCO C1(OC)CN(C(C2CC2(C)C)=O)CC1C(=O)NC1(CC2CCC2)CC1 C(=O)(CC(C)C(C)(C)CC)N1CCN(C(C(CC)=CC)=O)CC(CO)C1 N1(C2CCN(C(C3CCCN(CC=CC(=O)OC)C3)=O)C2)CCCN(CC)CC1 C(=O)(CC(C)C(=O)NC1CCC(C(=O)N(CC(C)C(C)C)C)CC1)OC N1(C(c2c(SC(C)C)cccc2)=O)CC(NC(C23CCOCC2C3)=O)CC(O)C1 c1(OCC(c2c(Cl)ccc(C(C)C)c2)=O)ccc(F)c(Br)c1F C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1C(NC(C(COC)C)=O)CC1 c1(OC)ccnc(O)c1C(N1CCC1CNC(c1ccnn1C)=O)=O CCC(C)(C(=O)N1CC2CC1C2CNC(=O)CC1(CO)CCOCC1)C(N)=O c1(SCC(=O)NCCn2cnc(C(=O)NC34CC(C3)C4)c2)ccccc1O N1(CC)CCOCC1C(=O)NC1CC1NC(c1ccc(=O)oc1)=O CCCCCC(C)C(=O)N1CCC2C1CCN2C(=O)CN1CCOC1=O Cc1cnn(CC(=O)N(CC(=O)NC(C)CC(N)=O)C2CC2)c1 CC1CCC=C1C(=O)N1CCC(OCCNC(=O)CC2CC(C(F)F)C2)C1 c1(OC)ccc(CN2CC(CNC(=O)CCCC(C)C)CC(F)(F)C2)c(F)c1F C(=O)(C(F)(CNC(=O)C(C(C)C)N(C(C)=O)CC)C(C)C)NCCCC C1(CC(=O)NCc2ccc(CNC(C3(O)COC3)=O)cc2)CC2(CCC2)CCO1 CCCC(O)C(CO)NC(=O)CN1CCN(C(=O)CC2CCCO2)CC1 C(=O)(CCCC(N)=O)N1CCC(COC2CCN(C(C(CCSC)O)=O)C2)CC1 C1(COC)(CNC(=O)CSC)CN(C(=O)CC(C)n2ccnc2C(C)C)C1 c1(CC(=O)NC2C3CCN(C(C4CC(CC)(CC)C4)=O)C32)ccc(F)c(C#N)c1 n1(CC)cc(C(N2CC(F)CC2CN(C(=O)C(C)C)C)=O)c2ccccc12 Cc1[nH]c2ccccc2c1CCNC(N1CCC(CC2CC2)CC1C)=O N1(C(C(=O)NC23CC(CNC(CCOCCOC)=O)(C2)C3)C)CCCCCC1 Cc1ccc(I)c(C)c1OCC(N1CCOC(CCCl)C1)=O N1(C(C(n2nnnc2C(C)(C)C)C)=O)CCC(N(C)C(C2(O)CCC2)=O)CC1 CCCC(O)C(CO)NC(=O)CC1CN(C(c2cnco2)=O)CCO1 CCCCC(C)(CO)NC(C1CCC2(CC2)N1C(=O)C=C(C1CC1)C1CC1)=O c1(C(C)OC)nc(C(=O)NCC(=C2CN(C(=O)CCc3cnc(O)[nH]3)C2)F)cs1 c1(NS(CC2ON=C(CC)C2)(=O)=O)nc(C)c(Br)c(C)n1 N1(C(C(CCC)(C)C)=O)CC(NC(c2occ3c2CCC3)=O)CC(F)(F)C1 CCC(C(=O)N1CCN(C(c2ccc(C)o2)=O)C(CC(F)(F)F)C1)C(C)C C#CCCC(O)CCNC(C1C2CCN(C(=O)C=CC3CCCN3C)CC12)=O c12nc(C)ccc1NC2=O.C1(C(=O)OCC)(C(=O)OCC)CC1C(F)(F)F.OCC C(C)(C)(CC(=O)NCCOC1CCN(C(c2cc(CO)ccn2)=O)C1)OC c1(C(=O)NC2C(CNC(c3n(CCCC)ncc3)=O)C2)cc2ccc(Cl)cn2c1 N1(C(COCCC(C)C)=O)CC2(CNC(C3CC4CC4C3)=O)CCC1CC2 c1(C(=O)NC2CN(C(c3nncn3C)C)C2)cc2sccc2s1 C1(NC(c2cc(C)nn2C)=O)C2CC3CN(C(=O)CCOCC(C)C)C1C3C2 N1(CCn2cc(CC(C=C)O)nn2)CCN(C(=O)CN2CCC(N(C)C)C2)CC1 n1(CC)nc(C(=O)NCC2(F)CCN(C(C3(CO)CC(C)(C)C3)=O)C2)cc1O Cn1cc(C(=O)NCC(CNC(=O)Cn2cc(C(C)O)nn2)CO)c(C(F)F)n1 C1(NC(c2cc(C)oc2)=O)CC2(C1)CC(C(=O)NC1CCCN(C3CC3)C1)C2 C1(C(N(CCC#C)C)=O)(CNC(C2CC3(CC3)C2)=O)CC12CCC2 N1(C(c2cnc(C(C)S(C)(=O)=O)[nH]2)=O)CC2CC1C2NC(=O)Cn1cc(C)cn1 N1(C(CC2C(C)CCN(C(=O)CC3CCSC3)C2)=O)CC2C(=O)NC(=O)C2C1 C1(CCCF)CCCN1CCn1cc(Cl)cn1 Cc1ncnc(C)c1CC(=O)NC1CN(C(C2CCCC3(CC3)C2)=O)C1 C(N=c1cc(C)[nH]cc1C(C)C)c1cn(-c2ccc(OC)cc2C)nn1 C#CCC(CCOC)N(CC(=O)NCCN(C1CC1)CC)C(C)C.OC C#Cc1cccc(C(c2nnnn2CC)Nc2ccc(C(F)(F)F)c(F)c2)c1 C(c1ccc(F)c(F)c1)=CC(=O)NC1CCN(C(CCCC=C)=O)C(C)C1 n1(CCCC)ncc(C(N2CCCC(N(C(=O)C(C)SCC)C)C2)=O)c1C C1(NC(COCCC)=O)C(C)CCN(C(=O)CCNC=O)C1C.C(=O)(N)NCC C1(C(N2C(CNC(C(N)=O)=O)CCC2)=O)COCCC1N.C1(CO)(CO)CCCCO1 C1(C)(CNC(C2(COC)CCOC2)=O)CCCNS1(=O)=O C(=O)(C(CC(C)C)N1CCCCC1=O)NC12CC(CNC(COC)=O)(OC1)C2 C(=O)(C(C)(C)C(C)(C)C)NCC(CNC(C(C(C)C)(C)O)=O)(C)C C1(C(=O)OC)(C(=O)NCC2CC(NCCN3CCC(O)CC3)CO2)CC=CCC1 c1(C(=O)OC)cc(CC(N2CC(F)(CNC(C3CCC3C)=O)C2)=O)ccc1O N1(C(C(C)SC)=O)CC(CNC(c2cc(Br)no2)=O)C(O)C1 Cc1cnc(C(=O)N(C)CC2CCCC2NC(=O)CC(C)N(C)C)c(C)c1 c1(C(=O)NCCCC(C)NC(C2CCN(C)C2)=O)ccc(C#N)c(Cl)c1 CC(C)C(CCN(C(=O)Cn1cncn1)C)N=c1nc(C#N)[nH]cc1Cl C=C(C)CC(C(=O)NCc1nccn1C1CC1)NC(=O)CCN(C)C c1(CNC(C)=O)ccc(C(=O)NC(C2(O)CCN(C(=O)C=CCF)C2)C)cc1 c1(C(=O)NC2CCCN(C(C3N(C(C)C)CCC3)=O)C2)cc(Cl)ncc1F c1(OC)cc(C(=O)NC(C)(C)CN(C)C(c2ccc(O)nc2)=O)cc(OC)c1O C1(O)(C(=O)NCC(C)CN(C)C(c2ccc(CF)cc2)=O)CCSCC1 c1(CC(=O)N(C(C)CCNC(=O)C=CC2CCC2)C)ccc(F)cc1C(F)(F)F C1(CC#C)(C(=O)NCCc2c(C)noc2Cl)CCN(C(=O)COC2CCOC2)C1 N1(C(C=COCC)=O)CCCC(CCNC(c2ncccc2N(C)C)=O)C1 c1(CC)ccc(S(=O)(=O)N2CCC(CN(C3CCN(C(C)C)CC3)C)C2)cc1 CC1CCN(C(=O)C=CC2CCCC2)CCN1C(C1CCCS(=O)(=O)N1)=O N1(C(C(C)(C)C2CCOC2)=O)CC2CCC(CNC(=O)CCF)(C2)C1 C1(C(N2CCC(NC(c3c(CC)nc(C)[nH]3)=O)C2)=O)CC2(C1)CC1(CC1)C2 Cc1cccn2cc(C(=O)NCC(C)(C3CC3)NC(=O)C3=CCCCCC3)nc12 C1(CNC(C(CC)C(C)C)=O)CN(C(c2nnsc2C(F)F)=O)CC(C)(C)C1 C(CCCC(C)NC(c1cc(C(F)(F)F)no1)=O)NC(c1cc(CCC)[nH]n1)=O c12ccccc1NC2=O.C(=O)(C(=O)NC(C)=O)C1C(C(=O)NCCN)C1.N(C)C C1(O)(C(C)NC(C2CC(c3cn(C(C)C(=O)N(C)C)nn3)(O)C2)=O)CCCCC1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(C(=O)OC(C)(C)C)C(F)(F)CC1.CC(CC#N)O c1(C(=O)NC2CCCC(NC(C(C)SC)=O)C2)cc(C)nc2c1c(C)nn2C CC(C)(F)CCC(=O)NC(C)(CNC(C1CCCCC(=O)N1)=O)CO C(=O)(C(C)C(C)NC(c1cccnc1O)=O)N1CC(OC)(CO)C1 C1(CC)C(NC(=O)C=CCN(C)CC)CCCN1C(C1COCCN1CC)=O C1(NC(CNS(N(C)C)(=O)=O)=O)CCN(C(c2cc(CF)on2)=O)CCC1CO c1(C[SH](F)F)cc(C)cnc1O.C(=O)(C(C1CCCC1)NC(=O)N)OC N1(C(Cc2cncc(C)c2)=O)CCC2(CC1)CC(NC(=O)C=CS(C)=O)CCO2 CCC(C)(C)CC(=O)N1CCCCC1C(=O)Nc1cc(CO)cc(F)c1 N1(C(C=Cc2n(CC)ccn2)=O)CCN(C(=O)Cc2ccc(C(C)=O)s2)CC1C c1(OC)noc(C)c1C(=O)NCC1CCCCC1C(=O)N(C)CCOC Cc1ccc(F)c(C(=O)NC2CCCCN(C(c3ccnc(O)c3F)=O)C2)c1O C1(CC(=O)NC(C2CC(NC(=O)COCCF)C2)C)OCCC1(C)C c1(SCC)c(C(=O)Nc2cccc(NC(c3cccc(F)c3)=O)c2)cccc1F C(=O)(CC(F)(F)C(C)C)NCC(CCNC(c1c(C)snc1)=O)O N1(C(c2c(CC)non2)=O)CCCCC1CCNC(c1oc(C2CC2)nc1C)=O c1(C(N2CC(O)(CNC(Cc3cn(CC)nc3)=O)C2)=O)cnc2c(ccn2C)c1 C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(=O)CC(=O)NC2CC2)C(C)C1 C1(C(=O)NC2CN(C(C3CNC(=O)N3)=O)CC23CC3)COc2cc(Cl)ccc2C1 N1(C(C(CCC2CC2)OCC)=O)CCC(CO)C(O)C1.C1(C)CCC(=O)N1 c1(OC)ncccc1S(=O)(=O)Nc1cc(-c2cc(C)ccc2C)ccn1 C1(O)(C(=O)NCC2N(C(c3scc(C)c3Cl)=O)CC=C2)CCc2ccccc2C1 CCC(C)(C(=O)NC1(CCNC(c2ccnc(C(F)(F)F)c2)=O)CC1)C(N)=O c1(OC)ccc(C(N2CCOCCC2C)C(=O)NCc2ccccc2)cc1I C(C1CCCN1C(C1CC1[N+](=O)[O-])=O)=CC(=O)NCCc1cocn1 c1(C(N2C(C)CCC2)=O)ccc2c(c1)CN(C(c1ccc3ncnn3c1)=O)C2 CC1Oc2ccccc2OC1C(N1CCN(C(c2cnsc2)=O)CC(C)(C)C1)=O C1(CNC(c2ccc(C)cc2F)=O)CN(c2ccnc(CSC)n2)CC(C)(C)O1 C1(COC)CC(CNC(c2c(Cl)cnn2C)=O)N(C(=O)C=C(C)C(F)F)C1 C(C(C(C)(C)C)NC(=O)CCSc1nnnn1C)NC(C(C)CF)=O CCC(C)(C(=O)N1CC(CC(C)NC(=O)CN2CCC(C(N)=O)CC2)C1)C(F)F C1(NC(=O)C2=COCC2)CCC2CN(C(=O)CO)CC2C1 C1(C(=O)OC)CCC(O)CN1C(c1cc(O)ncc1F)=O CC1OCCC1(C)OC(=O)NC(=O)NCC1CC(n2ccnn2)C1 c1(N2CCC(C(N(C)C)=O)C2)ncnc2c1ncn2CC(C)(C)C(O)C1CC1 N1(C(=O)NC2C=CC(Nc3cccc4[nH]ccc34)C2)CCc2ncccc2C1 C12(C(=O)OC(C#C)=O)CCCC(C(=O)OCC)(COC1)C2 c1(C(=O)NCC23OCC(CNC(c4c(CC)ccs4)=O)(C2)C3)cccc2ncnn12 C(=O)(CC(C(F)(F)F)c1ccccc1)N1C(C(C)(C)CNC(=O)CC#N)COCC1 C(CC(F)F)(C(=O)NCC(C)CC1CC1)NC(C(C)CN(C)C)=O c1(SCCC(N2CC3C(CNC(=O)C4=NOCC4)(C3)C2)=O)nc2ccccc2s1 c1(NC(C2CCCCCN2C(=O)Cc2ccco2)=O)ccc(Cl)cc1O C1(NC(c2ccc(OC)c(C)c2)=O)CCCCN(C(c2cnco2)=O)CC1 C(C)(C(=O)NCC(C)(C)n1cccn1)(C1CCCC1)NC(C(C)N(C)C)=O N1(C(CCN(C)CC)=O)CCN(C(=O)C(c2ccc(Cl)cc2)=O)C2CC12 c1(C(N2C(C(C)NC(c3cncc(N)c3)=O)CCCC2)=O)cc2cccnc2s1 c1(SCNC(=O)C(c2cncnc2)N2CCCC2CF)ccccc1I C1(C)(C(N(CCOC)CCNC(=O)CCCSC)=O)CC(C#N)C1.CC=C c1(C(N(CC)CC2CCCN2C(c2cc(C(=O)OC)on2)=O)=O)cc(OC)ccn1 c1(OC)cc(C(=O)NC(CCN(C(=O)C2=CCC2)C)C(C)(C)C)c(N)cc1F C(CCC(C)(C)C(=O)N1CC(O)C1)NC(c1nc(CC)sc1)=O c1(C(N2CC(OC)(CNC(C3CC(F)(F)C3)=O)C2)=O)cc2cnccc2o1 C1(C(N2C3CC(N(C)C)C3CC2)=O)CC2(C1)CC(F)C2.C12CC(=O)N(C1)C2=O C1(NC(C2CCCCN(C(c3c(NC)nccc3)=O)C2)=O)CCc2c[nH]nc2C1 C(N=c1[nH]c(=NCc2ccc(C)cc2)c2cc(OC)ccc2[nH]1)C1CN(CC)C1 CC(C(=O)N(C)CCNC(=O)CCOCCN(C)C)N1CCCC1 C12(C(N3CCC(NC(CCCC=C)=O)(CF)C3)=O)CC1Cc1c[nH]nc12 C(=O)(C(CC(C)CC(C)(C)C)N1CCCS(=N)(=O)CC1)NCCCSC c1(C(=O)NC(C)CNC(=O)C(F)=CC2CC2)cc(N)cnc1Cl C1(NC(CC(C)(C)C)=O)C(C)CN(C(c2cccc(C3(C#N)CC3)c2)=O)CC1C C=CC(C)CCC(=O)NCCC1(O)CCN(C(C2(CC)CC(C)(C)C2)=O)CC1 Cn1cc(C(N2CC3CC3(CNC(=O)COc3ccccc3F)C2)=O)ncc1=O C1(C(C(=O)NC(CC#C)(C)C)C)CCN(C(c2cnc(Cl)n2C)=O)CC1 C12(C(N3C(C(=O)OCC)CCC3)=O)CCCC1CCN2C(=O)CCC1CCCC1 C1(O)(CNC(C(n2nnnc2C(C)(C)C)C)=O)CN(C(c2n[nH]cc2C2CC2)=O)C1 c1(N2C(c3ncn(C)c3)COCC2)cccc(S(N)(=O)=O)c1[N+](=O)[O-] C1(C(=O)NCC2CC(NC(=O)COCC3CCCO3)C2)CCC(F)(F)C1 C1(NC(C2N(CC)CCC2)=O)CN(C(C23CC4CC2C3C4O)=O)CC1(C)C Cc1nn(C)c(C)c1CC(=O)NC1CC1NC(=O)C=CC(C)(C)C C1(OCC(N2CCN(C(C(c3n(C)nnc3)(F)F)=O)CC2)=O)CCC2(CC1)N=N2 CC1CCCC1CC(N1CC(=C(F)CNC(c2scnc2C2CC2)=O)C1)=O C1(c2cn(CCC=C(C)C)nn2)CN(C(c2cc(C)c(C)nn2)=O)CCN1C c12ccc(cc1)C(=O)OCC2.C(C)(CC(C)(C)C)OC(C=CC)=O C12(C(=O)NC3CC(CNC(C4(N(C)C)CC4)=O)C3)CCCCC1OCC2 N1(C(CN(C(=O)Cn2nnnc2C)CCOC)=O)CCC12CCC(O)CC2 c1(C(=O)NC2C(NC(C3CC(=O)NC3)=O)CCCC2)occ2c1CCC2 N1(CC(N2CC(OCCC(=O)OC(CC)C)C2)=O)CCC(C)CC1 N1(C(C(CC=CC)CC)=O)CC2(CCCC2)C1C(=O)NCc1cccc(O)n1 C1(C(=O)NCc2cc(C)ncc2)N(C(=O)C(C2CCOCC2)F)CC12CCCC2 C1(C(=O)Nc2cnc(O)nc2O)CCC2(CN(Cc3ccc(F)c(F)c3)C2)O1 CC1(C)Cc2ccccc2C1NC(=O)NCc1ccc(C2CCCCC2)cc1 CCC(C)(O)C(=O)N1CC(O)(CNC(=O)CCCc2cccc(Cl)c2)C1 C(=O)(C(C(C)C)n1cncn1)N(CC(C1CCCC1)NC(CC)=O)CC c12cc(ccc1C(F)(F)F)NC(=O)C2N(C)C.c1(CC)ccccc1F Cc1cc(C(=O)NC2CCC2NC(=O)C(C(C)C)Sc2ccccc2)nn1C C1(C(=O)NCC2(O)CN(C(C3CN(S(CC)(=O)=O)C3)=O)C2)CC=C(C)CC1 CCC(CC(=O)NCCc1ccncc1F)NC(C1CCCC1)=O c1(C(=O)NC2CN(C(c3c(OC)ccc(OC)c3)=O)C2)ccc2c(c1)COCO2 CC1CC(C(N2CCC(C(=O)NC(C)(C)CC3CCCC3)CC2)=O)CCO1 CN1CCC(=CC(=O)N(C2CCC(NC(c3cc(F)n[nH]3)=O)CC2)C)CC1 C1(C(N2CC(OCCNC(CCCOC)=O)C2)=O)CCCOC1c1cn(C)nn1 N12CCC(C1)N(C(=O)COCCO)CCC2=O.C1(OCCCOC)CC=CC1 C(C(C)(O)CC(=O)N(CC(C)CNC(=O)CCc1cccnc1)C)OC N1(C)CC(C)(C)C(C)C1.C(=O)(CS(N)(=O)=O)N1c2ccnc(n2)NCCC1.CCO Cc1ccc(C(N2CC(O)CC2CNC(=O)Cc2ccon2)=O)c(Br)c1 c1(C(N2CCC(NC(CC3C(C)CCCC3)=O)C2)=O)c[nH]c2cccnc12 C1(CC(=O)NC2CN(C(COCCCOC)=O)CC(O)C2)CCC2(CCC2)CO1 C(CCCCCNC(=O)CC1CC1C(F)(F)F)N(C)C(C1(O)CC1)=O C(=O)(CCS(=O)(=O)C(F)(F)F)N(CC(CC)NC(C1CCSC1)=O)CC C(CCC)(C(=O)N1CCCCC1C(C)(C)CNC(C1CCCC1)=O)=CCC N1(C(c2ccc(CNC(=O)CC3CC(F)C3)s2)=O)CCC(C2CC2)C1 N1(C(COCCCC#C)=O)CCN(C(c2oc(Br)cc2C)=O)CC1CCC C1(N(C(C(=O)N(CC(=O)OCC)CCC)=O)C2CC2)CCCOC1C CCC(C)(CNC(=O)C(CCOC)NC(=O)CC1C(=O)NN=C1C)CC c1(C(=O)NC2(CC(=O)NCCCN(C)C)CCC2)cc2cccnc2[nH]1 c1(C(N2CCC(CC#C)(C(N3CCC3C)=O)C2)=O)cccc(F)c1O C1(NC(c2ccnc(F)c2)=O)CC2CN(C(=O)CC3CC4CC4C3)CC12 c1(C(=O)NCCC2CC(NC(C3(COC)CCOC3)=O)C2)ccc(C#N)nc1O c1(CC(=O)NCC(C(C)C)(C)NC(c2cnoc2)=O)cc(Br)cc2c1OCC2 c1(OC)cncc(C(N2CC(CNC(=O)CCc3ccnc(Br)c3)C2)=O)n1 CC(C)CCCC(=O)NC(C)CCCCNC(=O)C(O)(C(F)(F)F)c1cn[nH]c1 C(N=c1[nH]cnc2cc(Br)ccc12)C1N(C(c2cc(C(C)C)[nH]n2)=O)CC(O)C1 c1(CC(=O)NC(CN(C(C(CC)OCC)=O)CC)C)c[nH]c2cc(Cl)ccc12 N1(C(C(CC)OC)=O)CC2CN(C(C3(c4cccc(Cl)c4)CC3)=O)CC(C1)O2 Cc1ccncc1CC(=O)NC(C1CN(C(c2coc(O)n2)=O)CCO1)C C12(C(N3C(C(=O)OCC)CCCC3)=O)CCCC1CCN2C(=O)CC=C(C)C c1(C(N2CCN(C(C=CC)=O)C(C)C2)=O)cc2cc(Cl)cnc2[nH]1 c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC2C)ccc2c(c1)C(C)CN2 c1(C(=O)NCC(CC)NC(C23CCCCC2C3)=O)c(C)ncn1C C(=O)(C1=Cc2ccccc2CO1)NCc1c2c(ccc1)N(C(COC)=O)CCC2 c1(C(=O)NCC(CN(C)C(C2(C)CSC2)=O)(C)C)cccc(C2CNC(=O)C2)c1 C#Cc1ccc(C(=O)NCCC2CC(NC(=O)CC(C)C(F)F)C2)cc1C c1(C(c2cccs2)C(=O)N(CCCC(F)(F)F)CC)cccc(Cl)c1 N1(Cc2n(CC)ncc2)CCC(C(=O)N(C2CSC2)C)CC1 c1(CN(C)C(C2(C)CCN2C(C2(C)CCC(=O)N2)=O)=O)cccc(Cl)c1 C1(NC(c2cc(CC)[nH]n2)=O)C2CC3C1C3C2C(=O)NCCc1cccs1 N1(C(C2CCCC(NC(C3CC(OC)C3)=O)CC2)=O)CCc2cncnc2C1 C=CCC(CNC(=O)CN1CCOCC1)C(=O)NCCCc1ccccc1C C1(C(=O)NC(CC(C)NC(=O)C(c2ccc(F)cc2)(C)C)C)CC1C1CCCC1 Cc1ccc2nonc2c1C(=O)NCCCC(C)NC(=O)CC1CC2CC2C1 C(C)(C)(CCN=C(NOC)NC1CC1c1c(Cl)cccc1Cl)C1CC1.C c1(CCC(=O)NCCCCC2CN(C(=O)CSC3CC3)C2)cccc(F)c1F CCCCCCCCC(C)CC(=O)NC(C)(CNC(c1ncc(F)cn1)=O)C1CC1 c1(NC(c2ccc(OCC)cc2F)=O)c[nH]c2c(C)cccc12 C1(O)(CC(N2CCC(C(C(=O)NC3(CCC)CC3)F)C2)=O)CCOCC1 CCCC(CC)CCC(=O)N1CCC(N=[N+]=[N-])C(O)C1 c1(C(N(C2CCCN(C(CCCOC(C)C)=O)C2)C)=O)cc2scnc2[nH]1 C#Cc1cccc(C(N2CC3CCC(C(=O)Nc4ccncn4)C3C2)=O)c1C N1(C(c2cc(C(C)=O)n(C)c2)=O)CCCC(O)(CN(C(=O)C2=NOCC2)C)C1 c1(C(C)=O)cc(C(=O)NCC(C)N(C)C(C2CC23CCCC3)=O)ccc1Br C1(C)(C(=O)NCCN(C(C(C2(OC)CCCC2)(F)F)=O)C2CC2)CCCC1O c1(N(CC(CSC)C)C)nc(C(F)(F)F)cc(=NC(C)Cc2ccccc2Cl)[nH]1 C1(C(=O)NC(C(C)C)CCNC(c2cn(C(C)C)nn2)=O)CNC(=O)CC1C N1(CC(=O)N(CCN(C2CCC2)C(C)=O)CC2CC2)CCOCC1=O C1(=CC(=O)NCCCCN(C(=O)C2=C(Cl)CCOC2)C)CC2CCC(C1)N2C C(=O)(C(O)C(F)(F)F)NC1CCC(F)(CNC(C2(C#C)CCC2)=O)C1 CC(C)(C(=O)NCC#CCNC(=O)C(F)(F)C1CCOCC1)C1CCOCC1 c1(N(CC)CC2CCN(C(=O)CCCF)CC2)cccc([N+](=O)[O-])c1C C(C(O)C(=O)N(C1(C)CC1)C)NC(COCC(=O)NC)=O C1(C(=O)NC(C=C)C)CC2(CC2)CN1C(c1ccc(OC)nn1)=O CC(C)CCCCC(=O)N(C(C)CN(C(=O)COCC(c1ccccc1)C)CC)C c1(N2CCC(C(C)C)C2)nc(=NCC(C)n2cccn2)[nH]c2c1CCCC2 C1(CC=C)(NC(c2nc(Cl)cs2)=O)CN(C(=O)Cc2cccnc2)C1 C(C)(CN=c1[nH]ccc(C#N)c1[N+](=O)[O-])NC(CCCOCCC)=O N1(C(C2CCCCO2)=O)CCN(C(c2cc(Cl)cnc2O)=O)C(C2CC2)C1 C=CC(O)(C(=O)NC(CNC(c1ccc(C2CCCO2)nn1)=O)CC)C(F)(F)F C1(C(CNC(C(C)NC2CCCC2)=O)C)CCS(=O)(=O)C1 Cc1cc(CC(N2CCC(NC(C3CCC=CO3)=O)CC2C)=O)cc(C)c1 c1(C(=O)OC)cccc(CC(N2CC(NC(=O)C(C)c3ccsn3)C(C)C2)=O)c1 c1(OC)cccc(C(=O)NCC#CCNC(=O)CC2(C(F)F)CC2)c1 Cc1cn(C)cc1C(=O)NC1CC(O)(CNC(c2cc(C(F)(F)F)ccn2)=O)C1 c1(C(=O)NCCCCN(C(C2(C#C)CCC2)=O)C)csc2c(F)cccc12 c1(C(N2CCC(CN(C(CN(C)C)=O)C3CC3)CC2)=O)ccc2c(c1)C(=O)NC2 CCCC(C)(CCC)C(=O)N1CCCC(CCNC(C2(OC)CC(C)C2)=O)CC1 CC(C)CCCC(C)C(=O)N1CC(C(C2C(OC3CCCSC3)CC2)=O)C1 N1(C(C2(C)CCCN2)=O)CCCC2(CCCNC2=O)C1.N12CCCC(CC1)C2=O c1(C(N2CCCCC(CNC(C3(CC#C)CC3)=O)C2)=O)c(C)ccc(Cl)c1N c1(OC)ccc(O)c(NC(=O)CC2C(NC(c3cnc(S)nc3)=O)CC2O)c1 n1(CC(=O)NCCN(C(C23CCC(CC2)C3)=O)CC)nc(C(F)F)n(C)c1=O C1(NC(C=CCOC)=O)COC2(CCN(C(=O)Cn3nc(C)c(Cl)c3C)C2)C1 CC1(NC(C2CC23CC3(F)F)=O)CCN(C(=O)CC=CCc2ccccc2)CC1 c1(OCC)ccccc1C(C)CC(=O)NC1CC(CNC(=O)C=CC(C)C)C1 C12(CNC(=O)CCc3cncs3)COCCN1C(=O)CN(C(=O)C1CC1)C2 C1(C(N(CCN(C(=O)CCN2CCCS2(=O)=O)C(C)C)C)=O)CC(=O)NC1(C)C c1(CCC(N2C(CN(C(C(CCC)C)=O)C)CCCC2)=O)ccc(Cl)cc1F Cc1noc(C)c1C(=O)NC1(CNC(C2CCN(C3CC3)C2=O)=O)CCC1 Cc1ccc(C)n1CC(=O)N(CCC(C)NC(=O)CC1CC2(CCC2)C1)C c1(C)cc(Cl)no1.N1(C(=O)OC(C)(C)C)CC(=CC(=O)OCC(=O)NCc2nc[nH]n2)C1 C1(CC=C)(C(=O)NC(c2nccn2C)C)CN(C(c2csc(=N)[nH]2)=O)C1 CC(C)C(CNC(=O)CC1CCCN(C)C1=O)C(=O)NCC#CCCO C1(OCC(=O)O)CCN(C(=O)NC2(COc3ccccc3)CCCOC2)CC1 Cc1nc(CC(N2CC(O)CC2CNS(=O)(=O)CC)=O)sc1C.n12cc(nn1)C2 CC1(C(=O)NC2CCN(C(=O)Cn3cnc(C(N)=O)n3)CC2F)CCCNC1=O C1(C)(CNC(CCOCC)=O)CCN(C(c2nn(C)cc2Cl)=O)CC1 N1(C(c2ncn(CC)n2)=O)CC(NC(=O)CNC(C)=O)CC(C)(C)C1 c1(OCC)nccc(C)c1NC(=O)C(O)C1CN(C(c2csnn2)=O)C1 CCCCC(C)CCC(=O)N1CCCC2(NC(=O)Cc3cccn3C)CCCC12 N(C(=NCCCF)N1CCCC(N2CCCCC2)C1)CCc1c(C)cc(Br)cc1 C1(N(C(CC(C)OC)=O)C)CC2CCC(C1)N2C(c1cnc(C(C)(C)C)[nH]1)=O C(=O)(CC(C)C(F)(F)F)NCC1(C)CCN(C(C2CC(OC)(OC)C2)=O)C1 CCCCC(C)C(=O)NC1(CNC(C2(F)CCOCC2)=O)CCCCCC1 c1(C(=O)NC2C(NC(C3C(C)(C)C3)=O)CC2)cc2c(cc1N)CCCC2 C(C1CCN(C(=O)C(F)C2CCC2)CC1)=CC(=O)NCCC1CCCC12CC2 CC1(C)CCCC(O)(C(=O)NC2CC3CCCCN3C2)CC1 c1(C(=O)NCC2C(C)CCN(C(=O)C(=O)NCC3CC3)C2)cc([N+](=O)[O-])cn1C c1(C(=O)NCCN2CCC(F)(C(C3SC(=N)NC3=O)C)CC2)cnc2ccccn12 N1(C(COCCCCC)=O)CCCC2(CCC(NC(c3cc(C)c(C)[nH]3)=O)C2)C1 Cc1cc(C(=O)NC(CNC(C2CCCS(=O)(=O)N2)=O)C(C)(C)C)cc(C)c1 c1(C(N(C2CCN(C(CC(=O)OCC)=O)C2)CC)=O)cc(C(C)C)nn1C C1(=O)C(C(C)O)N1.C1C(C)(NC(C)=O)C=CC(CC)=CC(=O)N1.CC=C C1(C(C(=O)N2CCC2CF)NC(=O)CCn2cccn2)CC=CCC1 CC1COc2ccccc2C1C(=O)N1CC(c2cnco2)C1 C12(CNC(c3cc(C(C)C)no3)=O)CCC(NC(=O)COC3(C)CCC3)(CO1)C2 C1(C(=O)NCC2(CO)CCCC2)C=CCCN1C(C1CCCC(=O)N1)=O C12(CNC(c3c(=N)[nH][nH]c3)=O)CCC(CC1)N(C(=O)CCSc1ccccn1)C2 C1(NC(C(C(CC)O)C)=O)CC2CCC(C1)N2C(C1CC1(c1ccccc1)C)=O Cn1nnc2cc(CNc3cn(C)c4cnccc34)ccc12 N1(CC=O)CCC(O)CC(C)(C)C1.C=CCC(C(=O)N1CCC(OC)C1)NC(C)=O N1(C(C(C(CCCC)O)C)=O)CCCC12CCCN(C(C1(COC)COC1)=O)C2 N1(C(Cc2nc(NC(C)=O)sc2)=O)CCN(Cc2nc(C3CC3)no2)CC1 c1(C(C2CC2)C2CC2)ccccc1F.N12CC(C(O)C1)NC(=O)C2=O C(CC(C)(C)C)N(C(c1cnn(C)c1)C)Cc1ccccc1 C1(NC(C(C2CCN(C(=O)C(C)(C)C)C2)C)=O)CCCCCCC1 CC1(C)CCCC(NC(C2CC(O)CN2C(c2scnc2Cl)=O)=O)C1 c1(CCC(N2CCC(SC(F)(F)F)CC2)=O)cccnc1F C(CCCC(=O)NCC(c1ccccc1)N(C(=O)C=CBr)C)OC c1(CNC(CC)CO)cccc(NC(c2cn(CC)nn2)=O)c1 C1(NC(CSc2n(C)ccn2)=O)CC2CC1CN(C(c1cn(CCO)nn1)=O)C2 N1(C(c2cnn(-c3ccccc3)c2)=O)CCC(C2(Nc3ncc(F)cn3)CC2)C1 C=CC(C)(C)C(=O)NCC(O)C(=O)N(C)C.C1C(=O)N1 C1(C(C(=O)OC(C)(C)C)NC(=O)NC2CCCC2F)CCCCCC1 N1(C(C(C)c2cccs2)=O)CCC(C(=O)N(C)CC2CCCS2)C1 C1(C(=O)NCCN2CCC(F)CC2)C2CN(C(=O)CC3CC3C(F)(F)F)CC12 N1(CC#C)CCN(C(=O)CSCCNC(c2ccncc2NC)=O)CC1=O C(=O)(CCCS(C)(=O)=O)NCC(N(C(C(C=C)c1ccccc1)=O)C)C1CC1 c1(C(N2CCC(NC(C(F)=CCC)=O)C2)=O)ccc(C2CC2(C)COC)cc1 C1(NC(=O)CSCc2ccccn2)CC2(C1)CN(Cc1cnccn1)C2 N1(C(c2n(C)cc(C#N)c2)=O)CCC(C2CC2)C1CNC(=O)CNC(=O)C1CC1 C(=O)(C1=NOC2COCC12)NCC(C)CC(=O)NC1CNC(=O)C12CC2 c1(C(=O)OC)sc2ncnc(N(CCCN(C)C(C3(O)CCCC3)=O)C)c2c1C c1(OC)cccc(CN(c2nnc(C3CCOC3)n2CCC2CCOCC2)C)c1 N1(C(c2cccc(C(=O)OC)c2)C(=O)NCC=C)CCCC1P(C)(C)=O N1(C(c2cnn(C(C)C)c2F)C(=O)NCCOC)Cc2cc(F)ccc2CC1C C1(C(N(C(CNC(=O)COc2cn[nH]c2)C2CC2)C)=O)CC(=O)NC(=O)C1 CCC(CC(=O)NCC(C)C(C)O)NC(=O)CC1(COC)CC1 C(CN=c1[nH]c2cc(F)ccc2o1)C1CCC(Nc2ccn3cc(C)nc3c2)C1 c1(OC)ccc(C(=O)C(N2CCC(O)(CNC(c3cc(C)on3)=O)C2)=O)cc1 CCCCCC(C)(C)C(=O)NCC(C)CN(C)C(c1cnn(C)c1C(F)F)=O C1(NC(C2N(N=O)CCC2)=O)COC2(C1)CN(C(C1CC(=O)C1)=O)C2 N1(C(c2c(C)cco2)=O)CCN(C(=O)C=CC(C)(C)C)C(c2nccn2C)C1 C12(CNC(c3c(CC)ncs3)=O)CC(COC)(CN1C(=O)C(F)C(C)C)C2 c1(C(=O)NCC2CCCN2C(c2sccc2C(F)F)=O)cnn2c(=O)cc[nH]c12 CC(C)CC(C(=O)N(C(C)(C)CC(=O)N(C)CC1CCCOC1)C)C(C)C c1(CCC)cc(C(=O)NCCc2cc(C(=O)NC3CC3C)no2)no1 CC1(C(F)(F)F)CN(C(C(CC2CCCO2)C(F)(F)F)=O)CCO1 c1(C(=O)OC)ncccc1NCc1cc(C)c(C(=O)NCC2(O)CCC(C)C2)o1 Cc1c(C(=O)NCC(C)NC(C2(C)CCCO2)=O)cccc1S(N)(=O)=O C1(CNC(c2[nH]cc(C)c2)=O)CC2(CCN(C(C3C(C)(C)C3(C)C)=O)C2)CO1 c1(NC(C(c2cccnc2)NC(=O)Cc2ccco2)=O)cccc([N+](=O)[O-])c1 C12(CNC(Cc3nc(C)[nH]n3)=O)COC(CNC(=O)CC3CCCC3)(C1)C2 C1(C(=O)NCc2c(OC)ccnc2)CCC(C)N(C(c2ccc(=O)n(C)c2)=O)C1 CCCCC(CC)C(=O)N1CC2CCC(CNC(c3ccnn3CCC)=O)C2C1 CC(C)S(=O)(=O)C(C)C(=O)NC1CC(C)(NC(=O)C=CC2CCCN2C)C1 C(=O)(NN1CCCC1C(N1CC(O)C(O)C1CO)=O)C1CCC(C)(C)O1 C#Cc1ccc(C(=O)NC(C)CCN(C(=O)C(c2cccnc2)O)C)c(F)c1 C1(C2CN(C(=O)Cc3ccn(CC(F)(F)F)n3)C2)(NC(CC(C)C)=O)CC1 N1(C(c2ccc(C(C)(C)C)cc2)=O)CC2CCC2(CC(=O)NC2CCC2O)C1 c1(OC)ccc(CNC(=O)C(c2ccc(Br)cc2F)(C)C)c(C)n1 Cc1cnc(Oc2cccnc2Br)c(C)c1 C(=O)(CC1OCc2ncccc21)NC1CN(C(c2cc(CC)no2)=O)CC1C C(CCCC(CO)NC(C1CC(=O)N(C(C)C)C1)=O)NC(c1cc(C)ncc1)=O c1(NC(CC2=CCCN(C(C3C(C(=C)C)OCC3)=O)C2)=O)ccc2nncn2c1 N1(C(C2CCC(C)CC2)=O)CC2CC1CN2C(C1(C)C=CCCC1)=O C12(C(=O)NCC34C(CN(C(c5ccc(C)cc5)=O)C3)C4)CC1COC21CCC1 c1(C(=O)NC2CC(C)(NC(c3n(C)nc(C(F)F)c3)=O)C2)ccc2cncn2c1 c1(C(=O)NC2C(CNC(C3(COC)CCOC3)=O)C2)cccc2nsnc12 c1(-c2cccc(CN3CCC4(C(C(=O)OCC)C4)C3)n2)cccc2c1OCO2 C1(CNC(=O)C=CSC2CCC2)(CO)CCN(C(C2CCCCCCC2)=O)CC1 C1(CCNC(=O)NC)CSCCN1C(=O)C(N1CCCCC1=O)C C(=O)(C(C(C)(C)O)NC(c1cc(C(C)=O)on1)=O)NC(C#C)C(C)C CC1(C)CCC(C(N2CC3(C(=O)NCc4nn[nH]n4)CC2CO3)=O)CC1 N1(C(Cc2ccc(C)o2)=O)CCCC(NC(C2(c3ccc(Br)s3)CC2)=O)C1C C(=O)(CC(CNC(C1CC(CF)C1)=O)C1CCC1)N1C(CN(C)C)CCC1 c1(C(=O)NC2(C3N(C(CCCC#C)=O)CCC3)CC2)cc2c(F)ccc(F)c2[nH]1 N1(C(C(COC)O)=O)CC2CC(NC(c3conc3C3CCCC3)=O)CC1C2 CC(Cc1ccccn1)C(=O)N1CCCC1CCNC(c1ccn(C)n1)=O C(=O)(C(CC(C)C)CC(C)C)NCC(CC=C)NC(=O)C(C)(C)NC(=O)NC N1(C(CCc2cc(C)no2)=O)CCC(F)(CNC(c2cc(C(N)=O)[nH]n2)=O)CC1 C1(C(=O)NCC2C(NC(c3ccc(C#N)[nH]3)=O)CC2)CCc2nncn2CC1 c1(OCCCC(N2C(CNC(CC)=O)C(C)CCC2)=O)nc2ccccc2s1 C(=O)(C(C)CCCC(C)C)NCc1cc(C(N(CCOC)CCO)=O)n[nH]1 Cn1nc2c(c1C(=O)NCC13CC1CN(C(c1cc(C(F)F)no1)=O)C3)CCC2 C1(OC)CC2CC(NC(=O)C(C)(C)C(C)NC(c3cncc(CO)c3)=O)CC12 S(=O)(=O)(CCCNC(C1CCCCN1C(=O)CCOC1CC1)=O)N(C)C C(=O)(CN=c1[nH]c(C)cs1)NC1C(OC)CN(C(C2CNC(=O)N2)=O)C1 N1(CC)CCN2C(=O)CCC2CCN1C(c1ccc2ccccc2c1Br)=O N1(C2CCCN(CC)C2)C(=O)NC(C2CCCO2)C1=O CS(=O)(=O)c1ncc(C(=O)NC2(CO)CCCN(C(=O)CO)C2)s1.C(COC)OC C=CCC(C)(C)C(=O)NCCC1(NC(=O)C2=COCCO2)CCC1 c1(CC(=O)NCC(CN(C)C(c2csnc2Cl)=O)O)ccc(C(N)=O)nc1 C1(NC(C#CC(C)C)=O)CC12CCN(C(C1C3COCC13)=O)CC2 N1(C(C2N(CC)CC2)=O)CCCCC(CNC(c2nn(C)nc2C)=O)C1 C1(C2CC(C)C2C)CCN(N2CC(CO)OC(C)(C)C2)C1 C1(CNC(C(C)NC(CC)=O)=O)CC2CCC1N2C(c1cccc(OC)c1N)=O C=CC1CC(NC(C2CCC(C(C)C)N2)=O)C1 Cc1cc(C)c(C(=O)NC2CCCC2CN(C(=O)C(F)C(C)(F)F)C)cn1 c1(NC2CN(C(C(CCC)C(C)C)=O)CC2SC)ccc([N+](=O)[O-])c(C)n1 Cc1cc(=NCCN2CCCC2=O)[nH]cc1S(=O)(=O)N1CCn2nnc(CO)c2C1 CCCC(C)(O)CC(=O)NCC(CNC(=O)C(C)(C)SC)S(C)(=O)=O c1(NC(CCC(C)(C)NC(C2CC2(F)F)=O)=O)cccc(N=[N+]=[N-])c1 C1(OC)(CNC(=O)C(C)(C)c2cnco2)CCN(C(=O)CSCC(N)=O)C1 C1(CCC)CN(C(c2ccnn2C(C)CC)=O)CCN1C(=O)COC(C)(C)CC c1(C(=O)NCC2ON=C(C)C2)ccc(CNC(=O)CC2CCCSC2)cc1 C=CC1(C(=O)NC(c2nccs2)CC)CCN(C(=O)C(CO)OC)C1 N1(C(C(=O)NCC2(C)CCCO2)=O)CC(F)CC1CC1CCOCC1 c1(C(=O)NC(C)CNC(C2CCC(=O)N2)=O)cc2ccc(Br)cc2s1 c1(C(C)NC(Cc2ccc(C)nc2)=O)nc2c(s1)CCC2 C1(CNC(C2C(CC(C)C)C2)=O)(CNC(c2cn(C)nn2)=O)CC(F)(F)C1 Fc1cc(F)cc2c1OCCCC2NCc1c(F)cccc1Br c1(C(N(C)CC2(NC(c3nc(OCC)oc3)=O)CC2)=O)cn2ncccc2n1 C1(CC(=O)N(C2CCOC2)CC)CCN(C(=O)CS)C1.C1(C2(C)CC2)CCCO1 N1(C(CCNS(CC)(=O)=O)=O)CCN(C(=O)CN2CCOC2=O)CC1CCO C1(NC(CCCCCOC)=O)CCC2(CC1)CC(NC(=O)CNC=O)C2 Cc1ccc(C(=O)NCC2CC2CC(=O)NC2CC(S(C)(=O)=O)C2)cc1O c1(C(=O)NC2CCCN(C(C(CC)C(C)(F)F)=O)CC2)noc2c1CC(C)CC2 C1(NC(c2c(C)[nH]cc2)=O)CN(C(=O)Cn2ccnn2)CC1C(F)F N1(C(C(C=C)O)=O)CCn2ncc(S(C)(=O)=NC(=O)C=CCC)c2C1 c1(C(=O)NC(C(=O)OCC)C)nn2c(c1-c1ccc(SC)c(C)c1)CCCC2 N(C1CCc2cc(F)c(F)cc21)Cc1c(-c2c(OC)csc2)ncs1 c1(N(C(CCCC)=O)c2nc(CC(=O)OCC)cs2)cc(C)c(C)c(C)c1 N1(C(C23CCC(OC)C2C3)=O)CCCC2C(NC(=O)CN(C3CCC3)C)C(C)(C)C12 C1(C)(C(N(CCCCCNC(C2CCN(C(CC)=O)C2)=O)C)=O)CCOCC1 c1(COC)nc(C)ncc1C(N1CC(O)(CNC(C2CC23CC3)=O)C1)=O c1(CC(=O)NCC(C(=O)N2CC(C(N)=O)(N(C)C)C2)OC)c(C)n[nH]c1C C(=O)(C(F)CCC(C)C)N1CCC2C(NC(CCOCCC)=O)C2C1 N1(C(=O)OC)CC2CC2(NC(C2(CC)CN(C(=O)CC3CCC3C)C2)=O)C1 C(=O)(C(CN(C(=O)OC(C)(C)C)CC)C(C)(C)C)NC1(C#C)CCNC1=O c1(CC(=O)NCC(CNC(=O)CCCCC2CC2)CO)cc(O)nnc1O C1(C(=O)NCC2CN(C(C3N(C(C)=O)CCC3)=O)C(C)C2)CC1C1CCCC1 Cc1cc(-n2cccn2)nc(=NCC2CC2(c2ccccc2)CO)[nH]1 C(=O)(C1=NOCC1)NC1(CCCCNC(c2c(CC)occ2)=O)CC1 N1(Cc2ccn(CC)n2)CCCC2C1CCN2Cc1cc([N+](=O)[O-])ccc1Br C=CCC(CNC(=O)COC)C(=O)N(C)CC1(OC(COC)=O)CCC1 C1(NC(c2cnc(C)n2C)=O)CCC12CN(C(=O)CC(=O)N(C)C)C2 CC(CS(C)(=O)=O)C(=O)NCC1CC1CNC(C1(C(F)F)CCCO1)=O c1(C(=O)NC(CNC(COCCCC#C)=O)C2CC2)ccc(OCCF)cc1 c1(NC(CC2(N(C)C)COC2)=O)cc2c(cc1CO)OCO2 Cc1nn(C)c(Cl)c1C(N1CC2CC2(C(=O)NC(c2cccnc2)C(C)C)C1)=O C#CC(CC(C)(C)C)NC(C1(NC(C23CSCC2C3)=O)CC(O)C1)=O N1(C(C(C)OCCC=C)=O)CC2CC(C1)CN(C(c1ccncc1F)=O)C2 c1(C(=O)NCC2CCC(F)(CNC(CCOC)=O)CC2)ncn2ccccc12 C1(CCNC(c2c(CC)ccs2)=O)CCN(C(C2CC(F)(F)C2)=O)C(C)C1 N1(C(COCCC#C)=O)CC(NC(=O)CCc2cncc(Cl)c2)CC(C)(C)C1 c1(CNC(C2C(C(=O)OC)C2)=O)cc(NC(=O)COCC2(C)CCCO2)sc1C N1(C(C2CN(C(C)C)C2)=O)CCC(F)CC1C(=O)N(C)CC1CC1 CCC(CC(F)(F)F)C(=O)N(CCCCNC(c1ccc(CN(C)C)o1)=O)C C#Cc1cccc(CC(N2CC(C(=O)N(C)CCN(C)CCO)C(C)(C)C2)=O)c1 c1(OC)ncc(C)cc1C(=O)NC1CCCC(CN(C(=O)C=C2CCC2)C)C1 C1(C(=O)NCc2cc(C)cc(O)c2)CN(C(=O)C=O)CCC1(F)F n1(CC(=O)NCC2(NC(C3C(C)(Br)C3)=O)CCCCC2)ncc2cccnc12 C1(N(C(=O)CCCc2ccncc2)C)CC2CCC(C1)N2c1nnccc1C#N N1(C(C=C(C)Cl)=O)CC2CCC(NC(=O)Cc3cnc(C)nc3O)CC2C1 C1(CC(N2C(CCCC)CCC2)=O)C2CN(C(=O)CC3CC3(C)C)CC12 C1(CC)CCCCC1OCc1cn(C(C)CNC(=O)Cn2cnnc2O)nn1 C(=O)(CCC(O)C(C)(C)C)NCCC1=CCN(C(C(C)(C)n2cccn2)=O)CC1 N1(C(COC(CC)C)=O)CC2CC1CC2NC(=O)CCCC1CCCC(=O)N1 CC(=O)CCCC(C)C(=O)N1CCC(N(C(C2CC2(Cl)Cl)=O)CC2CC2)C1 N1(C2CCN(C(C(CC)SC)=O)C2)CCN(C(=O)C(C)(C)OCC(F)(F)F)CC1 C(C)(CCC(=O)NCC1(C)CC1(F)F)NC(CSCC=C)=O N1(C(=O)C(O)C2CC2)CC2CCN(C(=O)Cc3ccoc3)CCC2C1 C(CC(=O)N=c1ccn(C(C)CC)[nH]1)N(C(CCC=CCCC)=O)C c1(C(N2CC=CCC2C(=O)NCc2cccc(O)n2)=O)ccc2c(c1)CC2 c1(OC)ncc(Br)c(N2CC3CC(NC(=O)Cn4cncc4C)C3C2)n1 N1(C(CC2(NC(=O)CC3CCOCC3)CC2)=O)CC(CO)C(C2CC2)C1 Cc1nc(NC(C)CNC(=O)CCN(CCO)CCO)cc(C2CC2)n1 C(=O)(C1=CCCCC1C)NC1C(OC)CN(C(=O)C(C(C)C)SC)C1 N1(C(=O)CC2CC(NC(=O)Cn3cccnc3=O)C2)CCCc2occc2C1 Cn1cnc2nc(N3CC(O)(CNC(=O)C(F)C(F)(F)F)C3)ncc12 c1(CN=C(NC2CCC(C(C)(C)C)CC2)NC2CCCCC2)ccc(Br)c(F)c1 Cc1nc(C(=O)NCC2CCC2NC(c2cc(C3CC3)on2)=O)c2ccccn12 C(=O)(CCCCC(F)F)NCCN(C(C)C)C(C1CCCOC1c1cn[nH]c1)=O c1(-c2nc(C3CCN(CC)C3)on2)ccc(F)cc1.N12CC(C)(C1)CNC2=O n1(-c2cc3cnn(C)c3cc2)nc(C2Cc3ccccc32)nc1C(O)C(C)(C)C C(C)(C(O)C(C)C)NC(c1c(CNC(C(C)OCCOC)=O)occ1)=O N1(C(Cc2nc(C)oc2)=O)CCCC(C(C)C(=O)N(CC2CC2)CC2CC2)C1 N1(C(c2c(Cl)ccc(OC)c2)=O)CCC2(CCN(C(c3ccc(C)[nH]3)=O)C2)C1 c1(C(N2C(C3CCN(C(C4(OC)CCCC4)=O)C3)CCC2)=O)cc(O)nc(O)n1 C#CCC(C)(C(=O)N1CCC(C)(COC)C1)NC(c1cccc(C)c1O)=O c1(CC(=O)NC(C)CN(C(=O)CC2C=CCCC2)C)cccnc1Br c1(CNC2CCC(NC(c3cscn3)=O)C2)ccc(O)nc1 CC(C)(C)C(C(=O)N1CCCC(O)C1)NC(C1CCCC(=O)N1)=O c1(C(=O)NCC2N(C(CCCc3n(C)cnn3)=O)CC(O)C2)n[nH]cc1[N+](=O)[O-] C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C)C(C1SCCS1)=O)(C)C N1(C(C2(COC)CCCO2)=O)CCOC(C)(CNC(c2csc(C)c2)=O)C1 O=NN1CCCC1C(=O)NC12CC(NC(C3(F)CCOC3)=O)(C1)C2 N1(C(c2cn(CC)nc2C)=O)CCC(NC(=O)CCC2(C)CC2)C(F)C1 CCCCC(CNC(C1CC(O)C1)=O)NC(c1cc(CC)no1)=O C(CCCCNC(C1CCCS1)=O)N(C)C(c1cc(F)c[nH]1)=O C12(C(=O)NC(C)CCCCNC(C3CCOC3C)=O)C3CC(CC13)C2(F)F c1(N2CC3(CCC(CNCCOC)O3)C2)ccc(C)c(S(C)(=O)=O)c1 c1(OC)c(F)cc(C(N2CC(N(C)C(c3nc(Cl)cs3)=O)C2)=O)cc1Br C(=O)(CCC(C)SC)N1C(Cn2cc(-c3cn(CCCCCC)nn3)nn2)CC1 C1(NC(C(C)N(C)C)=O)CCC2CN(C(c3cnoc3)=O)CC2C1 C#CCCCCCC(=O)N1CC(C(O)C(=O)NC2CC3CCCC3C2)C1 c1(C(N2CC(CC(C)(C)CNC(c3cccs3)=O)C2)=O)cnc(O)c2cncn12 C1(CC)CN(C(=O)CNCSS(C)(=O)=O)CCN1C(=O)COC.C(C)(C)(C)OC(=O)N C1(Cl)(C(=O)NCC2N(C(C(CC(C)C)C)=O)CC(C)(C)C2)CC12CCOCC2 C1(C(=O)NCC2CN(CCC)C2)CCN(C(=O)CCC(=O)NC)C(CC)C1 N1(C(c2c(OC)nccc2)C(=O)NCCCc2cccc(F)c2)CC2(CCCC2)C1 N1(C(COCC=C)=O)CC(NC(C2(CO)CC(F)(F)C2)=O)CC12CCOCC2 CC1CN(C(=O)C(CO)c2ccccc2)CCCN1C(=O)C=Cc1ccccn1 c1(CN(C(=O)OC(C)(C)C)NC(=O)CCNC(C)CC)nccn1C C#Cc1ccc(C(=O)NC2CCCC(N(C)C(c3coc(C)n3)=O)C2)cc1F Cc1nc2ccc(C(N3CCC4CN(Cc5ccc(I)c(O)c5)CC34)=O)cc2[nH]1 N1(C(C2(C)CCNC2=O)=O)CCN(c2ccnc(C#N)n2)CC(C)(F)C1 C12(NC(=O)C=CC3CCOCC3)CCOCC1CN(C(C1(Cl)CC1)=O)C2 c1(C(=O)NCCC2CN(C(CCC(=O)OCC)=O)C2)ccc2ccnc(O)c2n1 C(C)(C)(CC(=O)NCC1(O)CCN(C(=O)CCC2(C)CCC(=O)N2)C1)SC C#CC1CN(C(c2cc3ccncc3[nH]2)=O)CCN1C(C1CN(C(N)=O)C1)=O C=C(CNC(c1ccnn1C(F)F)=O)CCNC(=O)CC1(C)CC1F CC1=NN(c2ccc(C(=O)NCC(F)CNC(=O)C3=CCC(C)CC3)cc2)CC1 c1(C(=O)NC2CCN(C(CCCC#C)=O)C2)cncc(C#N)c1 c1(C(=O)NC2CC(C)(C(=O)NC3CC4CC4C3)C2)cn2c(n1)CCC2 CC(Cc1cccc(F)c1)CC(=O)OC(C)(C)COCCO.C1(C)CC1 CC1(C)CCOC(C(=O)NCC(=O)NC2CC(C)(C)OC2=O)C1 C1(NC(c2cccc(CC)c2)=O)CCN(C(c2ccnn2C(F)(F)F)=O)CC1F C1(CC)CCC(C(=O)NC(C2CN(C(=O)C(O)Cc3cn(C)cn3)C2)C)O1 CC1CC=C(C(=O)N2CC3CC(C2)C3CNc2ncnc3scnc23)CC1 C1(CCCCC)CCCN(C(c2ccc(CNC(C)(COC)CC)o2)=O)C1 C12(CN3CCCC(CNCc4scc(C(N)=O)c4)C3)CC1CCC2(F)F C(=O)(C(C)C(O)C(C)C)NCCCOCCCNC(CC(CCC)C)=O Nc1ncc([N+](=O)[O-])cc1C(=O)NC1CCC(NC(C2CCCN2C=O)=O)CC1 C1(NC(C(F)=CCC)=O)CC2(CCCCN2C(c2cccc3c[nH]nc23)=O)C1 c1(CNC(CC2C(C)C2)=O)ccc(N)c(Cl)n1.C12(CCCC1)C(=O)NC2 N1(C(C)=O)CC(O)CC1C(=O)N(C1CCCN(C(C2CCCO2)=O)C1)CC1CC1 C1(CNC(c2cc(CC)on2)=O)CC2(CC2)CN1C(=O)C(COC)NC(C)(C)C N1(C(C2(OC)CCCC2)=O)CCC(CCN(C)C(C2CCCCC2F)=O)CC1 c1(N(C(=O)C(=O)NCCCN)C)ccnc(CNC(c2nscc2Br)=O)c1 C1(CNC(C(N)=O)=O)CC2(CCOCC2)CN1C(=O)CC1CCCOC1 c1(N2CCC(N(CCC)C(c3ncsc3Br)=O)C2)ccc(C#N)nn1 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCC(CN(C)C(C2(C3CC3)CC2)=O)C1 Cc1ncnc(C)c1C(=O)NCC(CO)NC(=O)CSc1nnnn1C1CC1 c1(C(N2C(C(C)NC(COC(CC)(C)C)=O)CCC2)=O)cc(Cl)cn1CC n1(CCCC)nnnc1C(C)(CSC(C)C)NC(C)CC1CCOC1 C1(C(N2C(CNC(CCCCCCC)=O)CCC2)=O)COc2ccc(F)cc2C1 C(=O)(C(C)CC(F)(F)F)NCc1c(C(=O)NC(CC)C2CC2)con1 N1(C(c2c(CNC(C3C(C)(C)C3(F)F)=O)ccs2)=O)C2CCCC1CC2 CC1C(N(C(=O)C(C)(C)C2CC2)C)CCN1C(=O)CC1(C)CC1 c1(C(N(CC(CC)NC(=O)C(C)S(N)(=O)=O)C)=O)cc2ncccc2[nH]1 c1(CC(=O)NC2C=NN(c3cccc(Br)c3)C2=O)ccc2c(c1)OCO2 Cc1cn2cc(C(N3CC4(CCN(C(C5(C)CCC(C)O5)=O)C4)C3)=O)ccc2n1 C(=O)(C1=CCCCC1)NC1CCC(C(N(C2(C#C)CC2)C)=O)CC1 N12CCN(CC1)Cc1cn(nn1)CCC2=O.c1(CC(C)SC)nc[nH]n1 C1(NC(CN(C(=O)CC2CCCSC2)CCOC)=O)CCCC(O)CC1 C1(C(=O)NC(CN(C(=O)CCCC(N)=O)C)(C)C)CC2(CCCC2)C1 C1(C(N(CCN(C(=O)CN2CCC2C)C(C)C)C)=O)COc2ccc(Cl)cc2O1 C1(NC(C(C)OCCCC)=O)CCN(C(=O)Cc2cnc[nH]2)CC1O C(=O)(CCCCC1C(=O)NCCCN1C)OC.c1(SCC)cnc(Cl)c(C)c1 N1(C(C(C)c2ccco2)=O)CCCC(F)(C(=O)NCCN2CCCC(O)C2)C1 N1(C(C(C)N2CCCC2)=O)CC2(CC(NC(=O)C(C)(O)C3CCC3)CO2)C1 c1(CN(C)C(C2(CC(F)(F)F)CC2)=O)ccccc1CNC(C1(C)CC1(C)C)=O CC1CN=NC(=O)CN1CC(=O)NCCc1ccc(-c2nn[nH]n2)cc1 O(NC(=O)COCCNC(c1ccoc1C1CC1)=O)C(CC)C CC(=O)CCCC(C)C(=O)NC(C)C(C)NC(C12CCC(CC1)CO2)=O C1C(C)(C)CC(=O)N1.c1(C(=O)NCc2ccn(C)n2)cccc(F)c1O Cc1ccccc1NC(C1CC1C(N)=O)=O.C(=O)(C(C(C)C)N1CCCCC1CO)N C(=O)(C#CC(C)(C)O)NC(C1CN(C(=O)C(O)c2ccsc2)CCO1)C O=S(=O)(C(F)(F)F)N1CCN(Cc2cnc(N3CCCCC3)nc2)CC1 c1(NC(C2OCCN(C(COCCOC)=O)C2)=O)ccc(Br)cc1COC Cc1ccc(C(=O)N(C)CCOCCCNC(c2cc(-c3cccs3)on2)=O)o1 c1(O)ccc2c(c1)CCCC2.C1(=O)CCC(=O)NCC2(CC2)CNC(=O)C1.CCN N1(C(c2n(C)cnc2)=O)CC=C(CC(=O)N2CC(c3nncs3)C2)CC1 C1(NC(C(CC)O)=O)(CNC(=O)Cc2ccc(C(C)=O)cc2)CCOCC1 N1(C(COc2cccc(C)c2)=O)CCC(CNC(C2(C)CC(F)C2)=O)C12CCC2 C(=O)(C(C)(C)CC1CCC1)N1C(CN(C(C(c2scc(C)n2)(F)F)=O)C)CCC1 C(=O)(C(CC)CC=CC)N1C(C(=O)NCCCC#C)C(C)C1 C1C(C)(C)CN(c2ccc(C(C)=O)nn2)CC1(C)C.CO C(C(O)C(=O)NOC(c1ccccc1)=O)NC(c1cccc(F)c1)=O Cc1ncc(CC(=O)NC(CNC(C2(c3cncnc3)CCCC2)=O)C2CC2)s1 C1(NC(=O)Cc2ccccc2)CC1C1CCN(C(c2ccc(Cl)cc2F)=O)CC1 c1(CN(C(c2cnc(OC)s2)C(=O)NCCOC)CCF)nc(C)c(C)s1 CC1CCC(C(=O)NCC2CCCS2)N(C(=O)C(C)OCCN(C)C)C1 N1(CC(=O)NCC(C)(CO)NC(CC)=O)C(=O)CC(C)(C)C1=O c1(OC)cc(F)c(C(N2CC(C)(NC(=O)CC3C=CCC3)C2)=O)c(Cl)c1 c1(CNC(CCC)Cc2nccn2C)ccccc1CO C#CC1CN(C(C2(C(C)C)CCN(C(=O)CCc3nncs3)C2)=O)CCO1 N1(C(C(C)OCCCC)=O)CCC2C(CCN2C(c2ccnc3[nH]ncc23)=O)C1 c1(C(=O)N(c2ccccn2)CC2CC2)csc(-c2ccccn2)n1 C1(CNC(C(COCC)n2cc(C(C3CCCC3)NC)nn2)=O)CCCCCC1 n1(CC(N2CC(CNC(C3(C#C)CCC3)=O)OCCC2)=O)cc(S(N)(=O)=O)cn1 N1(C(CC(C)C)=O)CC(NC(c2cc3c(s2)CCC3)=O)C2CCCC2C1 c1(C(N2CCC(CCC(=O)NC(C3C(C(=O)OC)C3)C)C2)=O)sc(O)nc1C c1(C(=O)NCC(CNC(C(C(=O)OCC)(C)F)=O)C)cccc2c1OCC2 C1(NC(=O)NCCc2cnc(C)s2)CC2CCC(C1)N2C(C)C Cc1nc(CC(=O)NCC2CC2NC(=O)COC2CCN(C)CC2)c(C)s1 c1(C(N2CC3C(CNC(CCOC(C)C)=O)(C3)C2)=O)cccc(Cl)c1C(F)F C1(C(=O)NCC2(CC)CCC(=O)N2)CN(C(c2ccsc2C)=O)CC1C1CC1 C1(C(=O)NCC2(NC(C(n3cc(Br)cn3)C)=O)CCOC2)CC2CCC(C1)O2 c1(SC)nnc(N2CCC(NCc3csc(C)c3)CC2)n1CC.S(C)(=O)(=O)CCl C1(NC(c2c(C)cc(C)[nH]2)=O)CN(C(=O)C=Cc2ccccc2)C2(CCOC2)C1 N1(C(c2cnc(SC)s2)=O)CC2CS(=O)(=O)CC2(NC(=O)C2=CCSC2)C1 c1(C(N2CCCC(N(C(C(CC)OCC)=O)C)CC2)=O)cn2cccc(C)c2n1 C12CCCC(C1)CNC(=O)C2.C1(C(F)F)(CO)CCN(C(=O)CC2CC2)C1 C1(C(=O)NC2CC(CO)C2)CC2CCC(C1)N2C(=O)Cn1ncccc1=O c12cc(ccc1F)NC2=O.CC(C)(C(=O)NCC(=O)NOCCCF)C1CC1 N1(C(c2cnn[nH]2)=O)CC(C2CCCN(C(C3CCC=CO3)=O)C2)C1 C1(CC(=O)NCCCCCN(C)C(c2ccsc2)=O)COc2ccccc2O1 c1(C(=O)NC2CC(N(C)C(C34CCC3C4)=O)C2)cccc(-c2ccc[nH]2)c1 CCC(C)C(=O)C(=O)N1CC2CC1C2NC(c1ccccc1)=O C1(NC(COC)=O)CN(C(=O)COc2ccc(SC)cc2)CC(F)(F)C1 N1(C(C23OCC(C(C)C)(C2)C3)=O)CCC2CN(C(C3(CCF)CC3)=O)CCC2C1 CCC1c2ccsc2CCN1C(c1c(N2CCCC2)ncnc1Cl)=O C(=O)(CC(C)P(C)(C)=O)NCC1(C(C)NC(c2c[nH]nc2C(F)(F)F)=O)CC1 Cc1ncc(Cl)cc1C(=O)NC1CCCCC1NC(c1conc1C1CCC1)=O c1(CC(=O)OCC(c2ccc(F)cc2)C)ccc(C(C)(C)C)cc1 N1(C(c2c(C)cn(C)n2)C(=O)NCCC2(C)CC2)CCC(C)CC(C)C1 c1(C(=O)NC2C3CN(C(C(C)C(C)(F)F)=O)CC32)cnc2nccn2c1 c1(C(N(CCNC(C(CC)n2cncn2)=O)CC2CC2)=O)cccc(C(C)C)c1 C(=O)(C1=CCCN(C(=O)Cc2ccn(C)c2)C1)N1CC(C)C(N(C)C)C1 CCC(C(=O)N1CCC(C2CCCN2C(=O)C=CCn2cncn2)C1)C(C)O C1(=CCNC(C2OCC(C)C2)=O)CCN(C(=O)CC2(C)CCCCC2)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCC(O)CN(C)C(C2CC(CF)C2)=O)c1Cl c1(C(=O)Nc2nc(C)c(-c3ccnn3C(C)C)cc2)cccc([N+](=O)[O-])c1 Cc1nc(N(C)C)sc1C(N1CCC(C(C)NC(=O)CCc2ccc(Cl)s2)C1)=O c1(CC(NC(=NC)NC(C)COCCOC)C#C)ccccc1Br C1(CC(=O)NC(c2nc(C(N)=O)co2)C)CCC(=O)NC1.c12nc(co1)C(=O)NC2 C1(C(=O)NCC(C2CCN(C(CC(C)(F)F)=O)CC2)(C)C)CC2C=CC1CCC2 C1(C(N2C(C(C)C)(CO)CCC2)=O)CCc2c(nnn2C)C1 c1(C(=O)NCC2CCCC2C(=O)NOC2CC2(F)F)cc[n+]([O-])cc1 c1(-c2nnc(N(C)CCN3CCOCC3)n2CCC#N)cc2sccc2s1 C1(NC(C(CCOC)C)=O)(CO)CCCN(C(=O)Cc2cccc(OC(C)=O)c2)C1 C1(CCC(N2CC(NC(CCC)=O)C2)=O)CCCCN1C(=O)CCOC1CCC1 c1(SCC(=O)N(CC(C)NC(=O)Cc2ccsc2)C)nnc(-c2ccccc2)o1 N1(C(CCCNC(N)=O)=O)CC(CNC(C2(C3CCCCO3)CC2)=O)C(O)C1 N1(C(CNC(C(C)(C)C)=O)=O)CCC(O)C(NC(C2OC3CCC2C3)=O)C1 N1(C(c2c(C)noc2C)=O)CCOCC(NC(=O)C=Cc2ccn(C)c2)C1 c1(OCC)ncc(C(=O)NCCC2(C)CCN(C(C3CCC3C)=O)C2)cc1Cl C(=O)(CS(=O)C(F)(F)F)NCC1(F)CCN(C(c2c(CC)cncc2)=O)C1 C12(CNC(c3c(COC)noc3)=O)CC(NC(C3CC3(C)C)=O)(CCO1)C2 C(C1CCCCC1)=CC(=O)NC(C(=O)NC(C(N)=O)C1CCCC1)C1CC1 C1(NC(C(C)NCCC)=O)CCC(CNC(c2cnn[nH]2)=O)C1.C12(CC1)C(=O)N2 CCCCS(=O)(=O)CC(=O)N1CC(NC(c2cc(F)ccc2Cl)=O)C(C)C1 N1(C(C=CC)=O)CCCN(C(=O)CCc2ccc(OC)c(OC)c2)CC1C C1(C(F)(F)F)(C(=O)NCC(CNC(c2cnn3c2OCC3)=O)O)CC2CCC1C2 c1(CCC(=O)NCCCCNC(C2C(OC)CC2)=O)ccc(F)c(F)c1 C1(C(N(C(C)CN(C)C)C)=O)CCN(C(=O)Cn2ccnn2)C12CCC2 c1(OCCC(=O)NC2CC2CNC(=O)CC2CCC2)cccc(C(N)=O)c1 c1(C(=O)NC(C)CC2CN(C(=O)Cc3cncs3)C2)cncc2nc(CO)[nH]c12 c1(CCC(=O)NCCCOCCN(C(C(C)C)=O)C)cccc(O)n1 C(=O)(CS(=O)(=O)C(C)C)N1C(C(C)C)CN(C(=O)CNS(N)(=O)=O)CC1 CCC1=C(C(=O)N2CCCN(C(C3CCCN(C(C)=O)C3)=O)CC2)CCCO1 C1(NC(C2(CC)CC2)=O)CCOC(CNC(C2CC3(CCC3)C2)=O)C1 CCC(CC(=O)NC1CC(NC(c2cc(C#N)c(O)nc2N)=O)C1)C(C)C C1(CNC(C(=C(C)C2CC2)F)=O)CN(C(c2ccc(N)c(N)c2)=O)CCC1(F)F C1(SCC2(C)C(CNC(=O)OC(C)(C)C)C2)CCCN(CCCO)C1 N1(C(C23CCC(OC)C2C3)=O)CC(NC(=O)C(C)OCC(F)(F)F)CC2(CC2)C1 NS(=O)(=O)c1ccc(F)c(C(=O)N(C2CCS(=O)(=O)CC2)C2CC2)c1 N1(C(C(c2ccccc2)C)=O)C2CCC1CC(N(C)C(C13CSCC1C3)=O)C2 C(=O)(C(C(=O)NCCC(O)C(=O)OC)OC)NC1(CCOC)CCC1 c1(C(=O)NCC(CNC(=O)CCn2cccn2)F)ccc(Br)cc1F CN(C)C(=S)NCC(=O)NCCCCN1CCCC1.c1(=O)ccc1=O.NC c1(NC(C2N(C(c3[nH]cc(C)c3)=O)CCC2O)=O)c(Br)c(C(N)=O)nn1C Cc1c(C(=O)NC2CCCCN(C(C3(CO)CCC3)=O)C2)nn(C)c1N C12(N3CCN(S(CC(C)C)(=O)=O)CC3)CCC1CN(C(=O)CCC(C)(C)F)C2 c1(CC)nn(C)c(CC(=O)NCC2(F)CC(NC(=O)C=CC=C(C)C)C2)c1Cl CC(CC(=O)NCCC1(C)CCCC1)C(C)(C)NC(c1coc(CO)c1)=O c1(C(=O)NC2C=CCN(C(c3c(OC)cccc3)=O)C2)cc(OC)cnc1F N12CCOCC(C1)NC(C)CCN=CC(C)C2=O.C(=O)(C(F)(F)F)OC CC(C)C(CN=c1ccc2nnc(-c3cccc(C(F)(F)F)c3)n2[nH]1)N(C)C C=C=C(C)CC(=O)N(CC)CC1CCN(C(=O)C(C#N)C2CC2)CC1 c1(NC(C2N(C(C(CC=C)OC)=O)CC(C)CC2)=O)ccc2c(c1)CCO2 N1(c2ncc(C)s2)CCC2CN(N2CC(C)Oc2ccccc2Cl)C1 n1(CC)c(C)cc(C(=O)NCCC2CN(C(=O)CCc3nc[nH]n3)CCO2)c1C c1(SC)ccc(NC(=O)NC2CCCN(Cc3cc([N+](=O)[O-])cs3)CC2)c(C)c1 C1(CC(=O)NCCCCOC(C)C)CN(C(C2COC(=O)N2)=O)CCO1 c1(C(=O)NC2C(NC(CSCC=C)=O)CCC2)cc(N2CCC(O)CC2)ccn1 C(=O)(C(F)C(C)(F)F)NC1CC(C(=O)NCCCN(C)C)C1(C)C O=C(CCC(=O)c1cccc(Cl)c1)NCC1(NC(=O)Cn2cnccc2=O)CC1 C1(NC(C2N(C)CCCC2)=O)COC2CN(C(c3scnc3Cl)=O)CC12 c1(C(N2C(C3CCN(C(c4cscn4)=O)CC3)CCC2)=O)cc2ncccn2n1 C1(NC(C2CC2(F)F)=O)C2CC3CN(C(c4cncc5ccccc45)=O)C1C3C2 c1(OC)cc(OC)c(OC)cc1NC(=O)N(C1CC2CNC1C2)CCCC(C)C Cc1ccc(C(=O)NCC(C)CNC(=O)C(C)N(C)C)c2cccnc12 N1(C(CS(C(C)C)(=O)=O)=O)CC2(C1)CN(C(=O)CN(c1ccncc1)C)CCO2 CCC(C)(F)C(=O)NC1CC(O)(CNC(c2cc(-c3ccco3)on2)=O)C1 CC(CCCO)NC(c1cn(C2(C(=O)O)CC2)nn1)=O C1(NC(CCCC#C)=O)CN(C(c2ccnn2CC2CC2)=O)CC12CC2 c1(C(=O)NC2C(NC(C3(OCC)CCOCC3)=O)CCCC2)ccc(F)c(Cl)n1 CCS(=O)(=O)c1ccc(C(=O)NC2(CNC(C3CC4CCC3C4)=O)CC2)c(N)c1 c1(C(=O)NCC(C(C)(C)C)NC(C23CC(F)(C2)C3)=O)cccc2ccnn12 c1(C(=O)NCCC(C(C)C)NC(C23CC(C)C2C3)=O)c[nH]c2nccc-2c1 C1(O)(C(=O)NCC(C2CC2)NC(C(C)c2ccsc2)=O)CC(C)(C)C1 c1(CNC(=O)COCC2CCC2)ccc2c(c1)CN(C(c1ccc(O)nc1)=O)C2 C1(CC(=O)NCCN(C(C=CCC)=O)CCOCCO)CC2C=CC1C2 C1(C2CCCCC2)(NC(C2C(C)CCN(C(C(CCOC)C)=O)C2)=O)CC1 CC1(C)CC(N)CC(C(=O)NCc2csc(-c3ccco3)n2)O1 C(=O)(C1CCc2ccccc21)NCC(C)NC(c1cc(Cl)cn1C)=O C1(CC(=O)NCCN(CC(C)O)C(C2C=C(C)CS2)=O)CC(CC)=NO1 c1(C(=O)NC(CC)CN(C(=O)COCCCCOC)C(C)C)cc[nH]c(=N)n1 N1(C(=O)CO)CC2CCN(C(c3cnc(N4CCS(=O)(=O)CC4)nc3)=O)C2C1 C(=O)(C(C#N)C(C)C)NC(C(=O)NC(c1c(C)nc(C)[nH]1)C)C(C)C c1(C(=O)NCC2N(C(C(CCC)C)=O)C3C(C2)C3)cnc2sccc2c1 C1(CC(=O)NC2(CC=C)CN(C(c3c(C)csc3Cl)=O)C2)CCCNC(=O)C1 C1(C(=O)NC2CCC(CCC(=O)NC3(C=C)CCC3)C2)CC1C1(C)COC1 c1(CCC(=O)NC2CC(C)(NC(C3C(=C)CC3)=O)C2)ccc(N)cn1 C1(C2COCCOC(=O)CN2)COc2ccccc2O1.c1(COC)ccccc1 c1(OC)ccc(Cl)c(C(=O)NC2CN(C(=O)C(C)CC(N)=O)C3(CCC3)C2)c1F CCC(C)(CNC(c1ccn(C(F)F)n1)=O)C(=O)N=c1ccn(CCOC)[nH]1 C1(NC(C2N(C(C)=O)CSC2)=O)CC(=O)N(C(C)C)C1.C12(CCCC1)C(=O)N2 N1(C(C(N2CC(C)C2)=O)C)CC2C(NC(=O)C3=NOCC3)C2C1 C(=O)(CC(C)CC(C)C)N1CC(C(C(=O)NC23CCC(C2)OC3C)OC)C1 C(=O)(C(O)CC(C)(C)C)NC1CC(NC(C(c2c(OCC)cccc2)(F)F)=O)C1 C(C(C)(F)CNC(=O)CNC(c1ccccc1)=O)NC(CN(CC)CC)=O N1(C(c2ccc(=NCC)[nH]c2)=O)CC(C)CN(C(=O)C(C)CSC(F)(F)F)C(C)C1 C1(CC)CN(C(=O)C(C(C)C)NC(=O)C(C)(C)CF)CC(=O)N1 C1(C(=O)NC2CCN(C(=O)CCCN3CCCC3)C2)CCCC2(C1)CC2(F)F n1(CC)ccc(CC(=O)Nc2csc(-c3ccc(C)o3)n2)n1 C1(C(=O)NCC2(NC(C(C)OC)=O)CCC2)CN(S(N)(=O)=O)C1 C1(C(=O)NC2CCN(C(=O)Cn3c(C)ccc3C)CC2C)(OC)CCS(=O)(=O)C1 c1(C(=O)NC(CCOCC)C)c[nH]nc1CCNC(C1CCCO1)=O c1(CN(C(=O)CCC2CCC(=O)N2)C)cc2nc(Cl)ccc2s1 c1(C(=O)NC(CNC(C(C)OCC#C)=O)CC=C)ccccc1CS(C)(=O)=O Cc1cc(C#N)cc(C(=O)NC2CCCC(NCc3ccc(N(C)C)cc3)C2)n1 c1(OC)ccc(C(N2CCCC(CC(=O)NC(C)Cc3cnccn3)C2)=O)nc1 c1(C(=O)NC2(CNC(c3c(C)n[nH]c3C)=O)CCOC2)ccc(S(C)(=O)=O)s1 C12(NC(C(=O)NC3CC(NC(CC(C)(C)C)=O)C3)=O)CCC(CO)(CC1)CC2 N#Cc1ccncc1C(N1CC(F)(C(=O)NCCN2C(=O)CSC2=S)C1)=O C(C(O)C(=O)N1CC(C(=O)NC2C=CCC2)(CC)C1)SC N1(C(=O)Nc2cc(Cl)cc(Cl)c2F)C2CCC1CC(N1CC(O)C(F)C1)C2 c1(C(N2C(C(=O)OCC)CC(C)(C)C2)=O)nc2ccccn2n1 C(=O)(C(C)(C)C(F)(F)F)OCC1N(c2ccc(OC(C)C)cc2)C2OCC(C1)C2 O(N(C(=O)NC1CCC(n2cc(-c3cnn(C)c3C)nn2)C1)C(C)C)CC c1(C(=O)NC2(CO)CN(C(Cc3cc(C)cc(F)c3)=O)C2)cnn2ncccc12 c1(OC)cccc(C(=O)NC2(CCCNC(C3CCCC3C)=O)CC2)c1F N(C1CCCOc2cc(F)cc(F)c21)C(=O)Nc1cccc(OC)c1.C1C(=O)N1 N1(C(c2c(CC)c[nH]n2)=O)CCCC(C2CCCN2C(=O)CO)C1 c1(OC)cccc(CCC(=O)N(CCCNC(=O)CC2(C)CC2F)C)n1 c1(C(N2CC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)cncc2cccnc12 Cc1nc(C)c(CNC(C2CCC(CNC(c3cccnc3C)=O)CC2)=O)[nH]1 CC1CCC(NC(=O)Cc2nccn2C)CN1C(c1ccc(C(F)(F)F)nc1)=O c1(C(=O)NC(C)CNC(=O)C=CC2(C)COC2)cc(N)cnc1Br n1(CCC#N)c(N2CCC(CCO)C2)nnc1CN1CCNC1=O N1(C(c2c(C)ncs2)=O)CC(NC(=O)Cc2cc(C)n(C)n2)C(F)C1 c1(NCC(C)C2CCC2)ccc(S(=O)(=O)NCC#CCCO)c(Cl)c1 C1(NC(=O)Cc2ccc(O)nc2)(CF)CCN(C(=O)Cc2ccccc2)C1 c1(C(=O)NC2CCC(F)(CNC(=O)Cc3cnoc3)C2)cc(F)c(Cl)cc1Cl C1(CN(C)C(c2ncsc2Br)=O)CCN(C(=O)C(=O)N(CC(F)F)C)CC1 N1(C(Cc2cccc(C(CC)C)c2)=O)CC2CCN(C(=O)C=C3CC3)CC2C1 CCC(O)CC(=O)N(CCC(=O)NC(CO)C1CC1)OC C1(C(N2CCC(N(C(CCC(=O)OC)=O)C)C2)=O)CCCC(C)(C)O1 N1(C(CNC(=O)NC)=O)CC2(CCC2)CCC1CNC(=O)COC(C)C C(=O)(CP(=O)(C(C)C)C(C)C)NCC(CNC(=O)Cc1ccc(F)cc1C)OC C(CC(C)C)(C(=O)NC1CN(C(=O)CCc2ccc(O)cc2)CC1C)OC c1(C(N2C(CNC(CC(C(C)C)OCC)=O)CCC2)=O)cccc(C#N)c1Br C1(NC(COCCCC)=O)CN(C(c2ncnc3c2CCC3)=O)CC(C)(C)C1 C=CCC(C)(C)CC(=O)NC1CCC(CNC(=O)C(CC)N2CCCC2=O)CC1 C1(NC(CN(CCC#C)C)=O)CN(C(c2ccc([N+](=O)[O-])n2C)=O)CC1C1CC1 C1(NC(c2c(C)cccn2)=O)CC2(CCN(C(=O)C=CCBr)CC2)C1 c1(N(C(c2cccc(CSC3CC4(CCC4)C3)n2)=O)CC)ccc(C)c(F)c1 c1(C(N2CCN(C(C3CCCS3)=O)CC2CO)=O)cc2ccc(Cl)cc2s1 C(CC(C)C(F)(F)F)C(=O)NC1C(C=C)COC1 c1(CC)nn(C)cc1C(N1CCC(C(=O)NC(C)C2CC2)(CF)C1)=O c1(C(=O)OC)ccc(C=C(F)C(N2CCC(C(N3CC(F)C3)=O)CC2)=O)cn1 c1(C(=O)NCC23C(CN(C(c4c(C)nc(CO)s4)=O)C2)C3)ccc(F)c(CO)c1 S(=O)(=O)(C1CC2(CC2)C1)N(CC(=O)N(c1ccccc1)C)C N1(C(COc2c(C(C)C)cccc2)=O)CC(C2(NC(=O)CC(C)C3CC3)CC2)C1 c1(C(N2CC(O)(C(C)NC(=O)CCc3nc[nH]n3)C2)=O)cncc(C(F)F)c1 C1(CNC(C(c2cnccn2)C)=O)CCCC2CN(C(C3(C4CC4)CC3)=O)CC12 CC1CN(C(c2cnsc2)=O)CC(C)N(C(c2ncnn2C2CCOCC2)=O)C1 Cc1cc(N)c(C(N2CCC(CNC(C3(n4cnnn4)CC3)=O)C2)=O)c(F)c1 CC(C)C(F)(CNC(=O)C(C)n1ccnn1)C(=O)NOC1CC2CCC1C2 c1(C(N2CCC(CCNC(C(C)N(C(C)=O)C)=O)C2)=O)cnc2onc(C)c2c1 c1(C2N(C(CCC3CCN(C(c4c(C)nc[nH]4)=O)C3)=O)CC2)c(C)noc1C C(=O)(CC(C(F)F)NC(=O)C(F)=CC1CC1)N1CCC(OC)C1 CCC(CCCC(=O)NCc1csc(C)n1)NC(=O)C(F)F Cc1ccc2c(c1)SC(C(N1CCC1CNC(c1cnc3nccn3c1)=O)=O)C2 n1(CCCCNC(N(CCCCCC)C)=O)c(O)nc2ccccc12 c1(OC)cc2c(O)nc(O)nc2cc1CC1=NOC2OCCCC12 c1(C(=O)NCC2CN(C(CC(C)(C)O)=O)C3C2C3)sccc1S(N)(=O)=O c1(OC)cnc(F)cc1C(N1CC(NC(=O)CCn2cc(C)cn2)CC(C)C1)=O c1(CC)cc(Cl)ccc1C(=O)NC(CNC(c1cnc(C(C)(C)C)[nH]1)=O)C1CC1 c1(C(CCOC)NC(=O)C(C)=C2CCCC2)ccccc1[N+](=O)[O-] C1(C(=O)NC(CCC=C)C2CC2)CCN(C(=O)Cc2ccn(C)n2)C12CC2 n1(CC)ncc(CC(=O)NCC2(CC3CC3)CC2)c1Br.C12(CC1)C(=O)N2 N1(C(C2CC(S(C)(=O)=O)(n3cc(CC)nn3)C2)=O)CCC12CC1(CCOCC1)C2 Cc1cn2c(=O)c(C(=O)NCC3CCC4(CN(C(=O)CC(F)F)C4)O3)cnc2s1 c1(C(=O)NCC2C3CN(C(C(C)C(C)(F)F)=O)CC32)cnn2ccn(C)c12 Cc1cc(C(c2nnnn2CCOC2CC2)NCCC2COC2)cc(Br)c1 N1(C(C(C)n2cccn2)=O)CC2(CCCN(C(C3(CF)CCC3)=O)C2)C1 C1(NC(C2CC2F)=O)CCSC12CN(C(c1cncc(-c3ccccn3)c1)=O)C2 Cc1cc(C)c(C(=O)NCC2CCCCN2C(c2cnco2)=O)c(O)c1 N1(CC)C(=O)NC(c2cc(Br)cc3[nH]c(COC)cc23)C2=C1CCNC2=O C1(CC(=O)N(C(CNC(Cc2cc(C)sc2C)=O)C)C)Cc2cc(F)ccc2O1 C1(N(C(=O)CC2CCOCC2)CC)CCCN(C(c2ccsc2)=O)C1 N1(C(CC(C)(C)C2CC2)=O)CC2CCC(C1)N2C(=O)CC1SC2=NCCN2C1=O C(=O)(C1CCCn2c(C)nnc21)N1CC2N(C(CSCC)=O)C(CCC2)C1 C(=O)(CCCCC(F)(F)F)NC1CN(C(CS(CC)=O)=O)CC(C)(C)C1 CCCCC(CC)CCC(=O)NCC1CC(O)CN1C(c1cc(C)cs1)=O C(=O)(C1=CS(=O)CCC1)N1CC(C)C(NC(c2nccc3ccncc23)=O)C1 C1(CNC(CCC)=O)CC2(CCOCC2)CN1C(=O)C(C)(C)CCC C1(C2CC2)(C(=O)NC2(c3ccc(C(F)(F)F)cc3)CC2)CCC1 C=CCCCC(C(=O)NCC1CCC(C)N1C)NC(=O)C(C)=C1CCCC1 c1(NC(=O)NC2C(C)COCC2)cnc(Cl)c(Cl)c1 C1(NC(C2ON=C(CC)C2)=O)Cc2ccccc2C1NC(c1ccccc1Br)=O N1(C(c2onc(C)n2)=O)CCOCC(CNC(C2CCN2C)=O)C1 CCCC(CCCNC(c1n[nH]c(CC)c1C)=O)NC(=O)C=CC1CCC1 c1(C(=O)NCC(C2CC2)NC(C(CC)n2ccnc2)=O)nc(=N)cc[nH]1 N1(C(CC)CC)CC(C(N2CCN(C(=O)CCc3c[nH]c(=N)[nH]3)CC2)=O)CC1=O CC(C)CC(C)C(=O)NCC=CC(=O)NC(C)C(=O)NCCF Cc1ccc(CC(=O)NCCCC2(NC(C3CCC(=O)N3)=O)CCCC2)s1 N1(C(C(C)n2cccn2)=O)CCOCC(F)(CNC(c2ccoc2Cl)=O)C1 C1(NC(C2C(C)(C)CO2)=O)CCCC2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 c1(C(c2n(C(CC)(C)C)nnn2)NCc2nn(C)cc2C)cccc(C)n1 CS(=O)(=O)CC(=O)NCC1CCN(C(c2cnc(-c3ccccc3)cn2)=O)C1 N1(C(c2cc(C(C)(C)C)no2)=O)CC2CC1CCN2C(=O)CC1(CO)CCC1 Cc1cccc(SCC2CC(CN(C)C(c3cc(C)c(Br)s3)=O)C2)c1 C1(CNC(c2cc(C)nnc2O)=O)N(C(=O)C(C)NC=O)CCCC1(C)C N1(CCC)C(CCN(C)C)(C(=O)NCC=CCCCCS)CCC(CCCl)C1=O Cc1ccc(F)cc1C(=O)NC1CCN(C(=O)C(n2cc(Cl)cn2)C)CC1C N1(C(c2c(C)snc2)=O)CC2(CCCC2)C1C(N1CC=C(CO)CC1)=O c1(COC)ccc2[nH]nc(C)c2c1.C1(C(=O)N(C2CCCCC2)C)(N)CCSC1 N1(C(c2nc(C(=O)NC3CC(OCC)C3)co2)=O)CCC(C)(NC(C)=O)C1 C1(C(N2CC(NC(C3CC(C(=O)OC)C3)=O)C(O)CC2)=O)CCn2ncnc2C1 c1(C(=O)NCCC(C)N(C(c2nc(CCC)oc2)=O)C)ncc2c(F)cccn12 C1(C(CNC(=O)OC(C)(C)C)NC(C2(F)CCOC2)=O)CCC(F)(F)CC1 C1(C)(NC(C(CCOC)NC(=O)CN2CCNC(=O)C2)=O)CCC(=O)NC1=O C(=O)(CC1CCc2cc(Br)ccc21)NCC(CNC(CSCCCC)=O)O Cc1ccc(S(=O)(=O)NC2CCN(C(c3cc4cccn4cn3)=O)C2)c(C)c1 CCC(CC)C(=O)N1CC=CC12C(=O)N(CC1CC1)C2.C(C)(C(=O)OC)OC S(=O)(=O)(c1cnc(C(C)C)s1)NC1CCN(C(c2ccc(OCC#C)cc2)=O)C1 C(C(C)C(=O)NCC(C1CC1)NC(c1cn(C)cn1)=O)OC c1(OC(C)C)cccc2[nH]c(C(=O)N(C)CC3(NC(C4C(C)C4C)=O)CC3)cc12 N1(C(C=CS(C)=O)=O)CCCC2(C1)CN(C(c1[nH]nnc1-c1ccccc1)=O)C2 C1(C(=O)NCC(C=C)(C)C)(CNC(C2CC(SC)C2)=O)CC12CCC2 N1(C(c2ccc(CC)[nH]2)=O)CCN(C(c2c(Cl)cnn2C)=O)C(C2CCCC2)C1 C(CCC(C)C(=O)N1CCN(C)CC1CNC(c1ccc(Cl)nc1C)=O)OC N1(CC2OCC(C)C2)CCC(=O)N(CCOC=O)C1=O C1(C(N(C(C)C(=O)NCC2(C#N)CCC2)C2CC2)=O)CCCC1(C)C c1(N(C)C)ccc(C(O)C(=O)NCC2CCCN2C(=O)C=Cc2cn[nH]c2)cc1 N1(C(C2(NC(N)=O)CC2)=O)CC2CCC1CN2C(=O)CN1CC2C=CC1C2 Cc1cc(C#N)ccc1C(=O)NCC#CC(=O)NCc1ncn(C2CC2)n1 C1(CNC(COCCCC)=O)CN(C(=O)C(c2ccc(Cl)nc2)(F)F)CC1(C)C C(=O)(C(C(C)(C)C)OC)N1CCC(OCC(=O)N(CC(C(=O)NC)C)C)C1 CCCC(C)(O)CNC(C1(C)C=CCN1C(c1cc(COC)on1)=O)=O N1(C(C2CCC(CC)O2)=O)CCC(C(=O)NCC(CO)C2CCC2)=C(F)C1 C1(C(N2C(COC)CN(C(=O)COCCCF)CC2)=O)CCc2c(nnn2C)C1 C12(CNC(CC(C=C)CC)=O)CCCC(CN(C(c3n[nH]c(C)c3C)=O)C1)C2 N1(C(C(C)OCC#C)=O)CCC(O)(CCNC(c2cccnc2C(F)F)=O)CC1 C(c1ccccc1)=CC(=O)NCCN(C(=O)CC1(C)CC1)CCOC Cc1cc(Cl)ccc1C(=O)NCC(CNC(c1cccc(C2CC2)c1)=O)CO c1(C(=O)NCc2ccc(C(N(C)Cc3nnc(O)o3)=O)s2)ccccc1C#N Cc1nc2ncccc2cc1CC(N1CC(O)CC1CNC(C1CC=CC1)=O)=O C(=O)(C#CC1CCCCO1)NCC(C)CNC(c1occ2c1CCOC2)=O C(CC(=O)c1ccccc1)(C(C)C)NC(=O)NCC.C12(CCOC1)C(=O)O2 CCCCCCC(CC)C(=O)NC(C)C(C)NC(c1conc1C(C)(C)C)=O C=C1CCN(C(=O)C(=O)NC(C2CCCCO2)CC)CC1(C)C c1(C(C(=O)N(C2CCC(NC(c3csc(Cl)n3)=O)C2)C)O)ccc(F)cc1 N1(C(CN(C(CCOCCC)=O)CC2CC2)=O)CCC(C(=O)O)C(F)(F)C1 C1(CNC(C(CC#C)C)=O)CCCC2(CN(C(c3c(F)cc(C)cc3Cl)=O)C2)O1 N1(C(c2n(CC)ccc2)=O)CCC(C(C)NC(c2cnc(C)n2C)=O)CC1 CC(O)C(F)(F)C(=O)N1CCC(NC(=O)C(c2ccn(C)n2)C)C(C)C1 C(c1cnc(C(C)(C)C)s1)=CC(=O)N(CCNC(=O)Cc1cnn(CC)c1)CC N1(C(C2CCN(CC)C2)=O)CC(C(N2CCC(CC(=O)NC)C2)=O)CC1(C)C C1(C(N(CCNC(CC2(COC)CC2)=O)C2CC2)=O)CCCC(F)(F)C1 C(C(CNC(c1cnnn1CC)=O)S(C)(=O)=O)NC(c1cncc(CC)n1)=O CC(C)CC(C(=O)NC1CCC(NC(=O)CC(O)c2ccccc2)CC1)N(C)C S(=O)(=O)(c1cnccc1NC1CCCc2occc21)NCC1OCCN(C)C1 N#Cc1cc2ccc1NCCNS2(=O)=O.c1(SC(N2CCCC2)CO)cccs1 N1(C(CC(=O)OCC)=O)CCCC2(CCCN2C(=O)C(C)CO)C1 C(c1ccc(Cl)nc1)=CC(N1CCCC(C(N)=O)C1)=O.CC1C(=O)NC1=O C1(C(=O)NCCC2CC(C(=O)O)C2)CN(C(C2CC3C=CC2C3)=O)CC12CC2 CC1CC(CS(=O)(=O)N2CCCC(C3CCCCO3)C2)=NO1 c1(-c2cc(F)c(C)c(F)c2)nc2c(s1)CC(C(=O)NC1(c3cnn(C)c3)CC1)CC2 N1(C(c2cc(C)[nH]c2C)=O)C(C(=O)NC(C)C(=O)OC(C)C)C2CC(O)C1C2 N1(C(=O)OC(C)(C)C)CCn2nc(C(N3CC(CO)CC4OCCC34)=O)cc2C1 c1(C(N2C(C(=O)NCCC(C=C)C)CSC2)=O)cccc(F)c1 N1(C(C(C)CC(F)F)=O)CCC2(CC1)CC(NC(C1(C)CCOCC1)=O)CCO2 N1(C(C(=O)N(C(C)C(=O)N(CC)CC)CCOC)=O)CCOC2(CCOC2C)C1 Cn1cc2c(CN3CCc4nc(-c5cccc(C#N)n5)sc4C3)cccc2n1 C(N=c1nc(N2CCC(C(F)F)C2)c2c([nH]1)CCS2)C1CC(=O)N(C)C1=O C1(C(=O)NC(c2nc[nH]n2)C)(C(C)C)CCCN1C(c1cncs1)=O C(C1=NOC2CN(C(C34CC(CO)(C3)C4)=O)CC12)NC(=O)Cc1ccccc1O Cc1ccc(OCCC(=O)NC2CN(C(c3ccncc3Cl)=O)CC2F)cc1C n12c3c(cc(cc3)c1=O)CC2.C1(C(=O)NCC(C)N(C(C)=O)C)COCCN1C c1(NC(N2C(CC)CCCCCC2)=O)cccc2c1NCCC2C C=CC1(C(=O)NCCc2cc[nH]n2)CCN(C(c2ccoc2CC)=O)CC1 c1(C(=O)NCCC2N(C(CCOCC)=O)CCCC2)ccc(C(C)C)c(C)c1 C1(CNC(=O)NC2C(n3cc(COC)nn3)COC2)Cc2cc(OC)ccc2O1 C(=O)(CCC(F)(F)C(F)F)NC(C)CC(C)NC(=O)CCCC1CC1 C(=O)(C(C)(C)CC(C)(C)C)N(CCOCCNC(CC(C)n1cccn1)=O)C N1(C(CCc2n(C)cnn2)=O)CC(C(=O)NCCCN2CCC(O)C2)C(F)(F)C1 c1(NC(=O)OC(C)(C)C)cc(NC2CCC3CC23)ncn1 c1(OCCOC)ccccc1C(N1CCC(CNC(c2nccnc2N)=O)C1)=O CC(C)(C#N)C(=O)N1CCC12CN(C(=O)OC1(c3ccccc3Br)CC1)C2 C1(C(N(C2CCCN(CC(=O)NC3CCCCC3(F)F)C2)C)=O)CCCC2(CC2)C1 C1(CC(=O)NC)CN(C(N2CCCC(OC)C2)=O)CCN1C(c1n[nH]cc1C)=O Cn1nc(C2CC2CO)cc1C(=O)NC1CCCN(C(=O)C(F)C2CCCC2)C1 C1(F)(CNC(COCC(=O)NC)=O)CCCN(C(c2ccccc2C(F)F)=O)C1 N1(C(CC2(C#C)CC2)=O)CCC2(CC1)CC2NC(c1cc(C)n(CCO)n1)=O N1(Cc2ccc(O)c(C)c2O)Cc2ccc(C(=O)NC(C)CO)cc2C1 Cc1cc(C(=O)NC2(CC(N3CCNC(=O)CC3)=O)CCC2)cc2c[nH]nc12 N1(C(Cc2c(C)nc[nH]2)=O)CCSCC1CCNC(=O)CC(F)(F)Br C12(C(=O)NCC(C)(C3CC3)NC(=O)C3=CCOC3)CCC(C(F)F)(CC1)C2 c1(C(=O)NC(C(CO)NC(c2cc(C)sn2)=O)C)cccc2c1ncn2C N1(C(CC2(C(SC)CO)CC2)=O)CCC(C)(c2cn(CCN3CC(C)C3)nn2)CC1 C(=O)(CCCCC(=O)N1CC(C2CN(C(=O)C(F)(F)C3(O)CCC3)CCO2)C1)OC CC(C)(C)C(C)(O)C(=O)N1CC(NC(=O)CCNC(=O)C=CCl)CC(F)C1 CCCC(C)(C)CC(=O)NC1CCN(C(=O)C(c2ccc(Cl)cc2Cl)O)CC1F c1(CNC2C(C(=O)O)CCN(C(=O)OC(C)(C)C)C2)cc2cnccc2[nH]1 N(C(=NCc1cc(Cl)cs1)NCC1CC1)Cc1cn(C(F)(F)F)nc1 C(=O)(C1CCCc2nc[nH]c21)N1CC(COC)(NC(=O)CN(C(=O)C(C)C)C)C1 Cc1coc(C(C)C)c1C(=O)NCC(C(C)(C)C)NC(=O)CC(C)C1CCCO1 CC1(C)CN(C(C2CC3CC2CO3)=O)CC1NC(=O)Cc1ccnc(O)c1 C(=O)(C1=NOC(C)C1C)N1CCC(N(CC#C)C(c2cn(C3CC3)cn2)=O)C1 C1(C(N2CC(C(C(=O)NC3CCC(O)C3)OC)C2)=O)(N(C)C)CCCCC1 CC1CC=Nc2c(NC(=O)C3CC3)cccc21.C123CCC(CC1)(C2)C(=O)O3 C1(F)(CNC(COCC)=O)CCN(C(=O)CN(C)CC)CC1 C1(C(C)C)(C(=O)NCc2cnc[nH]2)CCCN1C(=O)CN1CCOCC1=O CC(O)C(C)(C)C(=O)NCCCN(C(c1cn(C)c(=O)cn1)=O)C1CC1 C=CC(C)(CCOC)C(=O)NCCC1(C(=O)NC2COC(C)(C)C2)CCC1 C1(NC(CN(C)C(=O)NC2(CC(F)F)CCC2)=O)CCC2CC1CN2C(C)(C)C C1(C)(NC(CCOCC#C)=O)CCC(CNC(=O)C(O)C(C)C)CC1 c1(C(N2CCC(C)(C)C2CC(N2CC(N3CC(O)C3)C2)=O)=O)c[nH]c2cnccc12 C1(C)(OCC(=O)NC2(CCOC)CCC2)CN(C(C2CCCOC2)=O)C1 C1(CNC(c2cc(COC)on2)=O)CC2(CO1)CN(C(=O)CC1(C)CCCC1)C2 Cc1nnc2ccc(NC(=O)C(=O)NCCC3CCCOC3)cn12 C(C)(N=c1[nH]c(=NC(C)c2ccco2)[nH]c2c1COC2)c1ncc(C)o1 C(=O)(CCCC(C)(C)NC(c1cc(O)cs1)=O)NC(CC)CCCOC C12(OC)CCC(C(N3CCCC(N4CCN(C)CC4)C3)=O)(CC1)C(=O)C2 c1(OC)ccc(Br)c(CN2CC(c3ncccc3Br)(O)C2)c1F c1(C(=O)NC(C2CCN(C(=O)CC#N)C2)C)ccc(Cl)nc1OC(F)F c1(C(=O)NCC2CC(NC(C3(COC)CCC3)=O)C2)ncccc1Cl Cc1ccc(C(=O)NC2CC2NC(=O)Cc2cccc(C)c2Cl)c(C(C)C)n1 S(=O)(=O)(CCNC(C1(OC)CCOC1)c1nnnn1-c1ccccc1)NC CC12CCOC(C(=O)NC3CC(CC(N4CC5CC5(CO)C4)=O)C3)(C1)C2 c1(OC)cc2nn[nH]c2cc1C(=O)NC(C)CCNC(c1n[nH]cc1[N+](=O)[O-])=O C1(NC(C)=O)CC2CC(NCc3cc(C4CCCC4)no3)CC2C1 C1(C(C(=O)N(C)Cc2cn(-c3ccccc3)nn2)F)CCCNCC1 C(CCC(C)C)(C(=O)N(CC(C1CC1)OC)C)NC(c1ccnc(OC)n1)=O CC(C(=O)N1OC2CCC1CC2)C1CCN(C(c2sccc2F)=O)C1 CC1Oc2ccccc2OC1C(N1CCOC(CN(C)C(C2CC2F)=O)C1)=O N1(C(C2C(C(C)C)C2)=O)CCOC2CN(C(c3cnccn3)=O)CC12 C1(Cc2c(C)[nH]c3ccccc32)CCC2(CCN(C(=O)CC(F)(F)Cl)CC2)O1 c1(C(=O)NC2CC(F)(CNC(CN(C)C3CC3)=O)C2)c(N)cc(F)cc1Cl c1(C(=O)NCCN(C(CCC(=C)Cl)=O)C2CCCC2)c(C)nc(C(C)C)nc1O c1(N(CC(CC)C)C)cc(Br)ccc1S(=O)(=O)N1CCS(=O)C(C)C1 C(C1c2ccccc2CN1C(C1CCC(F)(F)CC1)c1nnnn1C1CC1)OC C1(C(=O)NC(CC)CNC(=O)CC2COC(=O)C2)CCn2nnnc2C1 S(=O)(=O)(C1CCN(C(c2ccccc2)=O)CC1)NC(C)Cc1ccc(Br)cc1 N1(C(C(C)=C2CCC2)=O)CCOCC1CCNC(=O)C(C)n1ccnn1 C(=O)(C1=COCCO1)NC1CCCN(C(CC#N)=O)C1 CCC(CC)(CC)C(=O)NCCCC(O)C(=O)NC1(c2ncccn2)CC1 Cc1c(-c2nc(C3CC3)nn2CCCO)cnn1CCO N(C(=NCCC)NC(C)COC(F)F)C(C#C)C C1(C(C)=O)CCN(C(c2nc(-c3cnccn3)no2)=O)CC1 c1(C(N(C2CC3CNC2C3)C(C)C(F)(F)F)=O)ccc2cncn2c1 C(=O)(N=S(C)(=O)C1CNC2(CCOCC2)C1)C1CCC(OC)CC1 N1(C(c2cn(C)nn2)=O)C2CCC1CC(CNC(C1(CN3CCCC3)CC1)=O)C2 C1(CNC(CCNC(N)=O)=O)CN(C(=O)CC2CCCCC23CC3)C2(CCC2)C1 c1(C(N2C3CN(C(c4c(C)cc(Cl)c(Cl)c4)=O)CC32)=O)ccc(C#N)c2[nH]ccc12 C1(C(=O)NC(C2CCN(C(C3(C)CCCS3)=O)CC2)(C)C)CCc2ccnn2C1 C12(CNC(CNC(CC)=O)=O)COCCN1C(=O)CN(C(=O)CCS(C)=O)C2 Cc1cc(C)c(C#N)c(NCc2ccc(C(C)CC(=O)O)cc2)n1 C1(C(CO)NC(c2nc(C)sc2)=O)CCN(C(C2CCC2C)=O)CC1 N1(c2ncc(C(=O)OC)cn2)CCC(NC(=O)CCC[N+](=O)[O-])C(O)C1 CC(C)C(C(=O)NCC(C)N(C)C(C1CCCOC1)=O)Oc1ccc(Cl)cc1 c1(N(C2CCNCC2(F)F)Cc2nc(C(C)C)sc2)ncnc2c1ccn2C N1(C(CCc2ccc(C(C)(C)C)cc2)=O)CC(NC(C2(F)CC2)=O)CC12CCC2 c1(C(=O)NCC(C)N(C(c2cnc(NC)cn2)=O)CC)cc2n(c1)CCC2 C1(NC(c2c(CC)scn2)=O)CN(c2cc(C3CC3)nc(Cl)n2)CC(C)(C)C1 C1(C(=O)NC(C(=O)NCC2C(N(CC)CC)COC2)C)CC(=O)NC(C)C1 CC1CC(C(=O)N2CCCC(C(=O)NCC3CC(=O)N(C)C3)C2)=NO1 c1(SCC(=O)NC2CC(NC(c3ncn(CC)c3)=O)C2)ccsc1[N+](=O)[O-] c1(C(=O)NCC(C)(CSC)OC)ccc(CCNC(C2CC(C)(C)CO2)=O)cc1 C1(C2CC2)(CNC(C(C)Cc2ccncc2)=O)CCN(C(C2(CCO)CC2)=O)C1 N1(C(c2n[nH]c(=N)s2)=O)CCC(CNC(=O)C(N2CCOCC2)C2CC2)C(O)C1 CC(CNC(=O)CC(C)(O)C1CC1)CN=c1[nH]c(C(F)F)nc(=N)[nH]1 c1(C(=O)NCC2(CNC(C(CC)C(C)O)=O)CC2)ccc2nccn2c1 C=CCC(F)(F)CNC(=O)CCC1(C)CN(C(c2cnn[nH]2)=O)C1 CC(F)(F)C(F)C(=O)NC1CCC(CCNC(c2ccccc2CO)=O)C1 N1(C(c2scc(C(C)=O)c2)=O)CC2CC(NC(=O)CCNC(N)=O)C(C2)C1 C1(CNC(C2CCC2(F)F)=O)CCCC12CCN(C(C1SCCS1)=O)CC2 C(=O)(C(C)(C)C(N)c1ccccc1)NCCC(=O)N(C(c1ccccc1)C)C CCC(C)CN=c1[nH]c(N2CCN3C(=O)NCC3C2)nc2c1CCCC2 N1(C(C(C)CNS(=O)(=O)c2ccccc2)=O)CC2CCCC(C1)C2O C(=O)(C(O)CC(N)=O)N(C)CC1C2CN(C(=O)CSCCC#N)CC12 N1(C(C(CC)COC)=O)CCN(C(=O)CC2(C)CC2(Cl)Cl)CC12CCC2 n1(CCC)cc(C(=O)NCC(C)(CO)NC(=O)CC(C)OC)nn1 CC(c1cccnc1)=CC(=O)NCC1CC(C)N(C(=O)C=CC2CC2)C1 C1(CCC=C)CCCN(C(=O)NC(c2ccc(Cl)cc2)C(C)(C)C)C1 CC1C(NC(c2cc(Cl)cn2C)=O)C(C)CCN1C(C1Cc2ccccc2N1)=O N1(C(c2nc(CCC)oc2)=O)CCSCC1C(=O)NCCCC1CCOCC1 C1(C(=O)NCC(CN(C(C2CCOC2C)=O)CC)(C)C)CC(=C(F)F)C1 C1(C(=O)NC2CN(C(c3c(CC)c[nH]n3)=O)CC(C)C2)CC2(CC(C)=NO2)C1 C(C(C(=O)NC1CCCC1N(C(=O)CCCCOCC)C)C(C)(C)C)OCC=C CC(C)CC(C)C(=O)NCCn1cnc(C(=O)NC2(C)CC(C)(C)C2)c1 c1(C(N)=O)ccc(C(N2CC3(CC3C(N3CCC3c3ccccc3Cl)=O)C2)=O)cc1 c1(N(C)C)cccc(C(=O)NCC2(NC(C34CCC(C3)C4)=O)CC2)n1 c1(CNC(CCSCCC)=O)ocnc1C(=O)OCC N1(C(C(CC)C(F)(F)F)=O)CCC2(CCCN(C(=O)CCC3CCCC3)C2)C1 Brc1ccc(-n2ncnc2CN2CCCCC2n2cccc2)cc1 C1(NC(C(C=C)O)=O)CC2CCC1N(C(c1ccc(C(F)(F)F)cn1)=O)C2 N1(C(c2c(C)nn(C3CCC3)c2)=O)CCCC2(NC(C3CCC(F)C3)=O)CC2C1 c1(OCC=C)cc(OC)ccc1C(N1CCCC1CN(C(=O)CC1CC1)C)=O c1(CC)nc(C(=O)N(CCCN(C)C)CCNC(c2cc(C(F)F)no2)=O)cs1 C(N=c1[nH]cnc2ccc([N+](=O)[O-])cc12)C1CC(NC(c2ccc(CCC)[nH]2)=O)C1 C1(C(C)NC(c2cc(CC)no2)=O)CCN(C(C2(C(F)(F)F)CC(O)C2)=O)CC1 CCCCCCCC(=O)N1CCC(C)(C)C1C(N1CC(=O)N(C)C(C)C1)=O CC(C(=O)NCCOCCOCCCNC(C1CCC1)=O)SC(F)(F)F C(CNC(C1(C(N)=O)CC1)=O)(C(C)C(C)C)NC(Cc1c(C)noc1C)=O c1(C(=O)NC2CCCC(CNC(C(C=C)(F)F)=O)C2)cc(C)c(Cl)c([N+](=O)[O-])c1 CC(C)(C)CCC(=O)C(=O)N1CCCN(CCNC(c2cn(C3CC3)nn2)=O)CC1 CC1CN(C(=O)CN(c2cnccn2)C)CCCN1C(=O)C1=CCCOC1 c1(C(N2CCC(C)C2CNC(=O)CC2CCC(=O)N2)=O)cc2cnccc2o1 c1(CC(N2C(C(C)NC(c3cn(CC)nc3)=O)CCC2)=O)c(C)cc(C)cc1C N1(c2nc(C(=O)OC)c(C)s2)CCC(C)(NC(=O)C(C)CF)CC1 c1(C(=O)NC(C)CNC(=O)C(C)(C)NS(C)(=O)=O)nnc(O)n1C C1(NC(=O)C(F)(F)c2cncs2)CN(C(C2(CC3CC3)CCC2)=O)CC1F N(C1CCCc2c1cnn2C(C)C)C(N1CCC(C)(N(C)CC)C1)=O C1(C(N2CCCC(N(C(=O)CCOC(C)C)CC)C2)=O)CC2(C1)CS(=O)(=O)C2 CCC(C)C(C(=O)NCCCCCCF)N(C(=O)CN1CC=CCC1)C CC1(NC(C2CC2F)=O)CN(C(=O)C(C)(C)c2cnc[nH]2)C1 c1(C(=O)NCc2nnn(CC)n2)cc2c(O)cccc2n1C CCCCN=C(NCCc1ccc(Br)cc1Cl)N1CCC(N2CCCC2)CC1 c1(C(=O)NCC(CC)(C)NC(c2cc(SC)oc2C)=O)ccc(P(C)(C)=O)cn1 c1(OC)ccnc(C(N2CC(CNC(=O)CC3CCCN(C)C3)C2)=O)c1O C1(NC(CCN(C(C)=O)C)=O)CN(C(c2ccc(Cl)s2)=O)CCC1C C#Cc1cccc(C(=O)NCC2CCN(C(C3(CCC=C)CC3)=O)CC2C)c1F c1(C(N)=O)cccc(C(N2CC(O)(CCNC(=O)C(F)(F)CO)C2)=O)n1 c1(N(C(=O)C(C)N(C)C(c2ccccc2C)=O)CC)ccccc1O c1(OCC)cccc(C(=O)NC2CN(C(c3sc(SC)cc3C)=O)CC2C)c1 C(=O)(N=S(C)(=O)C1CC(CN)C1)C1(C(=O)Sc2ccc(CC)cc2)CCOC1 c1(C(N2CCCC(N(C(C(CC)F)=O)C)C2)=O)ccc(F)c2c1OCC2 N1(C(C2(CC=C)CCN(C(c3ncoc3C)=O)C2)=O)CCCCC(F)(F)C1 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCN(C(c2cncc(F)c2Cl)=O)C2CC12 CC(CC(=O)NC1(C(=O)N(C(C)C(N)=O)C)CCN(C)C1)C(C)(C)C C(C1CN(C(=O)CC2CCCOCC2)CC1C(=O)NC1C2COCC12)=CC C1(CNC(=O)CCc2ccsc2)CC(N=c2[nH]c3cc(Br)ccc3o2)C1 N1(C(C2CC(=O)CN2C(C2OC3CCC2C3)=O)=O)CCC(CO)C(O)C1 Cc1cc2[nH]c(C(=O)N(C3CCCC3)NC(C3(C)CC4CC4C3)=O)cc2o1 C(=O)(CCC(=O)NCCOCCCNC(=O)C(c1cscn1)N(C)C)NCC c1(C(=O)NCC(CNC(C2C(C)(C)OCC2)=O)F)ccc2[nH]c(=N)sc2c1 Cc1cc(NC(c2conc2CNC(c2cnc(C)s2)=O)=O)cc(Cl)c1 N1(C(C(C)SCC2CCCO2)=O)CCN(C(=O)CSc2c[nH]c(=N)s2)CCC1C S(=O)(=O)(c1cccs1)NCC(=O)NC(CC)CNC(C1(C)CCCN1C)=O N1(C(=O)CCOc2ccccc2)CCOC2(CCCN(C(C3CCCO3)=O)C2)C1 CC1(CNC(=O)CC2CNC(=O)O2)CCCN(C(=O)Cc2nnc(O)s2)C1 Cc1ccccc1OCCC(=O)NCC1C2CC1N(C(=O)Cn1ccnn1)C2 c1(C(N2CC(OC)C(NC(=O)CNc3nc(C)cs3)C2)=O)cc(C)c(F)cc1N C#CCCCCCCN=C(NCc1ccccn1)NCC1CCOC1C(=O)OC Cc1cc(C)c2[nH]c(=NC3CC(O)(CNC(=O)CC4CC4C)C3)sc2c1 C1(CNC(CCCCC)=O)CC2(CCN(C(C3COC3)=O)CC2)CO1 CN1CC(C(=O)NCC2CN(C(C3C4CCC(F)(F)C34)=O)C2)OCCC1=O c1(N2C(CNC(c3cnc(F)c(F)c3)=O)CC(C)(C)C2)ncnc(Cl)c1[N+](=O)[O-] c1(C(=O)NCCC2(C(=O)NCc3c(C)cco3)CCC2)cc(N)cc(F)c1 c1(CN2C(C(=O)Nc3cc(C)cc(O)c3)CC(F)(F)C2)cccc2ncccc12 N1(C(C(C)n2cccn2)=O)CCC2(CC(NC(c3cnc4cc[nH]c4c3)=O)C2)C1 n1(CC(=O)NCCN(C(C2CCC(F)C2)=O)CC)cc(N)cn1 C1(C)(C(N(CCC(=O)NC(C2CCC2)C)CC2CC2)=O)CCCO1 c1(NC(C)=O)ccc(NC(c2ccc(-c3c[nH]nc3C)o2)=O)cc1Cl N1(C(C2CCC(=C)CC2)=O)CCCC(O)(CCNC(c2cnn(C)c2CC)=O)C1 C1(NC(Cn2cnc(=N)[nH]2)=O)CCOCC1NC(c1cnc(C2CC2)nc1)=O CC(C)(C)C(Br)C(=O)N1CC2(CC(c3ccccc3)C2)C1 C1(CC(=O)NC2C(NC(CC3(C)CCC3)=O)CCC2)C=CS(=O)(=O)C1 C1(C(=O)NC(CN2CCCS2(=O)=O)C2CC2)COc2ccc(F)cc2C1 c1(C(N)=O)ccnc(C(=O)NC2CC(NC(C3CCC(=O)O3)=O)C(O)C2)c1 C1(NC(c2nc(COC)oc2)=O)CC2C1CCN2C(=O)CSc1cccc[n+]1[O-] C1(CNC(C(C)N(C(=O)CC2CCC(=O)N2)C)=O)CCC(=O)N1 c1(OC)cc(C=CC(=O)NC(CNC(c2ccccn2)=O)C(C)(C)C)ccc1F C(CC)(CCS(C)(=O)=O)NC1C(CCCCCC)CCC1 c1(OC)ccc(-c2nnc(COc3ccccc3C(F)(F)F)o2)cc1 C#CCCC(O)C(=O)N1CCCC(CCNC(=O)Cc2csc(COC)n2)CC1 C(=O)(CC(CN(C)C)C(F)(F)F)N1CC(C)C(C)(CNC(c2cnsc2)=O)C1 C12(CNC(C3CC(C)C3)=O)CC(NC(=O)CN3CCOCC3)(CCO1)C2 c1(C(=O)NCCN(CCOCCO)C(C2(C)CC(=O)N(C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl S(=O)(=O)(c1c(NCC2CCC(N)CC2)cnn1C)N1CCCC(C(C)C)CC1 c1(NCC(C)N(C(=O)Cn2nnc(=N)[nH]2)C)ccnc2c1cnn2C c1(OCCC)cc(Br)ccc1CNC1CCCN(c2cc(C(C)C)ncn2)CC1 c1(NC(CC)=O)cc(Cl)cc(C(F)(F)F)n1.C12CN(CC1F)C2=O c1(C(=O)NC23CC(CNC(CC4(OC)CCCC4)=O)(C2)C3)ccc(C)c(F)c1N c1(OCC)ccc2cc1-2.c1(OC(=O)CCc2ncco2)ccc(OC)cc1 c1(C(N2CCC(CNC(=O)Cn3nnc(=O)[nH]3)C2)=O)cnccc1C(F)(F)F C12(NC(c3c(OC)cccc3)=O)CCCC1(F)CN(C(=O)C(C)N(C)C)C2 N1(C(c2cc(C)c(C)o2)=O)CCCC(C)C1CNc1nccnc1F n1(CC)nc(C2CC2)cc1C(N1CC2CC2(CNC(=O)CCS(C)=O)C1)=O N1(C(C(C)OCC=C)=O)CCCC(C)(C)C1CNC(c1ccc(=O)oc1)=O C(=O)(CC1OCCc2ccsc21)NCCCCNC(=O)CC1CCS(=O)(=O)C1 C#CCCCC(C)C(=O)Nc1cccc(NC(=O)C(CO)OC)c1 c1(C(=O)NC2C(SC)CN(C(=O)C=CC3CC3)C2)ccn2ccccc12 n1(CS(N2C(C(=O)NC(C(=O)OC)(C)C)CC(C)C2)(=O)=O)cnc2ccccc12 Cc1cccc(C(C)(C)C(=O)N2CCC(CNC(C3CN(CC(C)C)C3)=O)C2)c1 C1(NC(c2cc(C)c(F)cc2)=O)CN(C(c2ccnnc2S)=O)C2(CCOC2)C1 S(=O)(=O)(c1ccccc1)NC1CN(C(C2CC2F)=O)C1 C1(C)(CNC(c2c(OC)c[nH]n2)=O)CCN(C(C2CCC(N(C)C)CC2)=O)CC1 C(=O)(CC(C)(C)CCOC)NC1C(C(=O)NC(CCC)C(F)(F)F)CCC1 c1(C(C(=O)NCC2CCCC2)NC(C)C)ccc(F)c(Cl)c1F C(=O)(N=c1cc(C2CCCCN2S(=O)(=O)CC2CC2)[nH][nH]1)c1c(OC)ccs1 c1(OCC)ccc(Br)c(C(C)Nc2cnc(CNC)nc2)c1 C1(C(=O)N(C2CCCCCC2)C)(OC)CCN(C(=O)CC2CN(C)C2)CC1 c1(CCC(C)C)cc(C(=O)NC(C)CNC(c2cnc(C(C)O)s2)=O)no1 C1(C2CCN(NC(C3C(C)C3C)=O)CC2)(C(C2CC3(C2)CC3F)=O)CC1 N1(C(CCN(c2ccc(CCC#N)cn2)C)=O)CC2(CCN2C(=O)CC#N)C1 C=CCCC(C)C(C(=O)NCc1ccc(F)cc1)N1CC(C(=O)OC)C(CCC)C1 c1(CN(CC(C)NC(C2CC2CC(C)(C)C)=O)CC)[nH]c2c(C)cccc2c1C C(=O)(C1=C(C)OCCC1)NCC1C=CC(NC(C2C(OC)CCCC2)=O)C1 C#Cc1cc(C(=O)NC2CCC(F)(CNC(=O)CC3(O)CCCC3)C2)ccc1Cl O=C(O)C(O)Cn1cc(C(N2C(CO)CC2CO)=O)nn1 c1(SC)ccnc(O)c1-c1nc(CC2CCC2)nn1C1CCNC1 C1(N(c2ccc(O)c(C(F)(F)F)c2)C(C(CCC)Cl)=O)COC2(CCNCC2)C1 c1(N2CC3CC(NC(C4CCC5C(C4)C5(F)F)=O)C3C2)ncc2ccccc2n1 C(=O)(C(=O)N=c1cc(C(C)(C)C)o[nH]1)NCC(CCC)N c1(C(N2CCC(c3cccc(F)n3)C2)C(=O)NCCOCC)cccc(Cl)c1 C1(CC(C)NC(c2c(C)occ2)=O)CCN(C(c2cnc(Br)s2)=O)CC1 c1(OC)ccc(C(=O)NC2C=CCN(C(C3CC3Br)=O)C2)c(OC(C)C)c1 N1(CC)CC(NC(=O)C(C2(O)CN(C(=O)Cc3cc(C)n(C)n3)C2)F)CCC1=O CC1(CO)CCN(C(=O)Cc2cc(C(=O)O)ccn2)C1 Cn1nnc2cc(CCC(=O)NCC3C(C)CCN3C(=O)CC=C(Cl)Cl)ccc12 c1(NCC(=O)NC2C(NC(C3CCC(OC)C3)=O)CCC2)ccccc1[N+](=O)[O-] N1(C(CCCCN(C)C(C2(C)CC(C#N)C2)=O)=O)CCCC2CCCC12 N1(C(C(C)CO)=O)CCN(C(=O)Cc2cnco2)CC(C)(F)C1 n1(C(C)C)cncc1C(=O)NCC1(O)CN(C(=O)Cn2nccn2)C1 C(=O)(CCCCCN=[N+]=[N-])NC1(C(=O)NCc2cnco2)C(C)(C)C1 c1(OC(C(=O)NC(c2nnnn2C)CCOC)F)ccc(F)c(Cl)c1 N1(C(Cc2ccc(C)nc2)=O)CCCC(O)CC1.C12CC1C(=O)NC2 Cc1ccc(CC(=O)N(C2CN(C(=O)C(O)C(F)F)C2)C)cc1C c1(C(N2CC3CC(NC(C4CCC(C)(C)O4)=O)C3C2)=O)ccc(F)c(F)c1O c1(C(N(C2CCN(C(=O)CCCCC3CC3)C2)CC#C)=O)ncc[nH]c1=O Cc1cc(CNC2C3CN(C(c4cc(F)ccc4I)=O)CC23)cc(Br)c1 C12(C(N3CCC(C#N)(F)C3)=O)CC(CCO1)N(C(c1ccc(O)cn1)=O)C2 c1(N2CC(C(C)NC(C(COC)C)=O)C2)nc(C#N)c(Cl)s1 C1(CNC(CC(C)(C)C)=O)N(C(C2CCCN(S(C)(=O)=O)C2)=O)CCC1(C)C C1(C(=O)NC(C)C=CC(N2CCC(C(F)F)C2)=O)(SC)CC(=O)C1 N1(C(CCN(C(C(COCC)(C)C)=O)C)=O)CCC12CCC(C)CC2 C1(CNC(c2c(C)cnn2C)=O)C2CCCC1N(C(C1CCCN1C)=O)C2 c1(C(N2C(C(CNC(C3CC(=C)C3)=O)(C)C)CCC2)=O)ccc(OC(C)C)cn1 C1(n2cc(-c3c(C)ncs3)nn2)CON(C(=O)C2CC(=O)N(C(C)(C)C)C2=O)C1 c1(C(=O)NC2(CO)CN(C(C3OCCC(C)C3)=O)C2)cc2nccnc2[nH]1 N1(C(C(C(=O)OC)C)=O)CCC2(CC1)CN(C(=O)CCC1C(=O)NN=C1C)C2 c1(C(=O)NC(C)(C)CNC(c2cccc(C3CC3)c2F)=O)ccc2snnc2c1 N1(C(C(COc2ccccc2)OC)=O)CCOCC1CNC(=O)CC1CCSC1 C(=O)(CC(C)(C)C(F)F)N1CCC(COC)C1CNC(=O)C1=CC2C=CC1C2 Cc1cc(C(N2CCCC(F)(CNC(C3CN(C)C3)=O)C2)=O)c(N)c(Cl)c1 c1(OC)cc(C(=O)NCC2CCCN2Cc2ccc(O)nc2Cl)cc(OC)c1C c1(C(=O)OC)cccc(C(=O)NC2(CNC(=O)CC3(O)CCCC3)CCC2)c1 c1(OC)cc(C(N2CCC(C)C2CNC(=O)CCC(N)=O)=O)c(F)cc1N c1(C2(NC(c3n(CCCCCC)nnn3)C3CCC3)CC2)ccc(Br)cc1F C1(NC(CCCC)=O)Cc2ccccc2C1NC(=O)CCCn1ccnn1 C(C)(CCC(=O)N1CCC(CCNC(=O)CCC(C)NC(N)=O)C1)SC C1(CNC(Cc2scc(C)c2)=O)CCC(C(=O)N(C2CC2)Cc2ccon2)CC1 c1(CN2CC(CNC(c3csnn3)=O)OCC2)cc(F)c(F)c(F)c1 N1(C(CCC2CC(NC(CSCC=C)=O)C2)=O)CCN(C)C(C2CC2)C1 C1(C(N2CC(C#C)(C(=O)NC(C)CSC)C2)=O)CCC=CCCC1 C1(C(=O)NCC2(CCNC(C(C)(C)C3CCOC3)=O)CC2)COCC(C)(C)O1 c1(C(=O)NCC2C(NC(c3c(C)nsc3C)=O)C2)cccc2c1CCOC2 CCCCCC(O)C(C)C(=O)NCC(C)NC(c1cc(C)sc1Br)=O C(=O)(C1=COCCO1)NCCOC1CCN(C(CCCOC)=O)C1 C1(NC(C2(N(C)C)CC2)=O)C2CC1N(C(=O)CCCn1ccnn1)C2 C(CCN(C(=O)C(CC=C)CC(C)C)O)(C(N(OCC)CC)=O)CCC N1(C(C(C)OCC#C)=O)CCN(C(=O)Cc2sc(C)nc2C)CC(O)C1 c1(CNCC2C(C)C(C)CN2C(=O)OC(C)(C)C)cc2ccccc2n1C C(=O)(CC(C(F)F)NC(=O)C(F)OC)NC1(CCOC)CCN(C(C)=O)C1 C(=O)(C(C)(C)C(C)(F)F)NC1C=CC(CNC(Cc2cc(C)[nH]n2)=O)C1 c1(C(=O)OC)[nH]c(=NC(C2=CCCCC2)c2nnnn2C)cc2c1ncn2C CCC#CCN=c1[nH]c(=NC(C)c2nc(O)n[nH]2)[nH]c2c1CCCC2 N1(C(c2onc(CC)c2C)=O)C2CCC1(CNC(=O)CNC(N)=O)CC2 C12(C(N3CCC(C(CC(=O)Nc4cncnc4)C)C3)=O)CC3CC(C(=O)N1)C2C3 C1(C(N2CC(CC(C)(C)C)C2)=O)CC2C=CC1N(C(=O)Cc1nc(=N)[nH][nH]1)C2 C1(C(N2CCC(OCCNC(=O)C=C(Cl)Cl)C2)=O)CC2(C1)CC(F)C2 [N-]=[N+]=NC1CCN(C(C2(F)CCCN(C(C3CC4(CC4)CO3)=O)C2)=O)C1 N1(C(C2(NC(C(C)=NOCC#N)=O)CCN(C)C2)=O)CCN(C)CC1CCO N1(C(C(C)CCO)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)Cc1ccco1 C(C(=O)NCCC(N1CCC2CC12)=O)(C(C)C)NC(COC)=O C(CC(=O)N(C)CC1CC(F)C1)N(CC=C)C(C1CCN1C(C)(C)C)=O c1(CCOC(C)(C)C(=O)N2CCC(NC(=O)OC(C)(C)C)C2)c[nH]cc(Cl)c1=O c1(CN2C(C)CCC(NC(c3cnco3)=O)C2)cc2c(cc1Br)OCO2 C=C1CC2(C1)CC(C(=O)N(C)CCNC(c1sc(Cc3ccccc3)nc1C)=O)C2 c1(C(c2nnnn2CCNC(C)=O)NC(CCC(=C)C)C)cc(C)cc(C)c1 N1(C(C(C)CC(F)(F)F)=O)CC(NC(=O)CCc2cccnc2)C(S(C)(=O)=O)C1 CC(C)CC1(C(=O)NCCNC(=O)CSC2CC2)CC1 c1(C(N(CC(=O)NCC(CNC(=O)C(F)=CCCF)OC)C)=O)cccc(Cl)c1 Cc1cc(CNC2CC2C(=O)Nc2cccc(Cl)c2Cl)nc2nccn12 N12CCN(CC1)C(=O)C1CCC(CC1)NC1C(C1)C2=O.c1(COC)ccccc1 c1(C(N(C)CCNC(=O)CN(c2ccc(Cl)nn2)C)=O)cnc2n1CCCC2 c1(C(=O)NC2(C(N(CC#CC)C)=O)CC2C)cnncc1O c1(C(=O)NCC2(CNC(C3(O)CCC(CC)C3)=O)CC2)nccc(C)c1N CCC(C(=O)N1CCC(C(=O)N(CC(C)(C)OC)C)C12CC2)C(C)C N1(C(CC(=O)NCC)=O)C2CCC1C(C)C(NC(C1CCCS(=O)(=O)C1)=O)C2 CC1CN(C(=O)CC2CCC(=O)NC2)CC1NC(=O)CCCn1cccc1 C1(CC(N2CC(O)(CC(=O)NC)C2)=O)CC(NC(=O)C=CCN(C)C)C1(C)C c1(C(=O)NC2(N3CCOCC3=O)CC2)nc2ccc([N+](=O)[O-])cc2s1 CC(C)CC(C(=O)N(CCF)C1CC1)N(C(=O)CCc1ccn(C)n1)C C1(C(N2CCN(C(c3ccc(C)cn3)=O)C3C2C3)=O)CC2CC(O)CC(C1)C2 c1(C(N2C(CCC)CN(C(=O)CCS(C)(=O)=O)CC2)=O)cnc2nncn2c1C N1(C(CCC)=O)CCCC2CN(C(C3CC(C)(O)C3)=O)CCCC12 C1CCCCNC(=O)c2cnn(c2)CC(=O)N1C(C)C.C1(C(=O)N(C)C)CC1F N1(C(C2CC(SC)C2)=O)CC2C(CNC(c3ccc(CS(N)(=O)=O)cc3)=O)C2C1 Cc1ccnc(C(N2CCC(C(C)(C)NC(=O)Cn3ccccc3=O)C2)=O)n1 C#Cc1cccc(C(N2CCN(C3CN(C(=O)C(C)c4ccsc4)C3)CC2)=O)c1 C1(NC(CC=CC)=O)CC2CC(NC(=O)Cn3c(C)ccc3C)CC2C1 Cc1cc(C)cc(C=CC(N2CC3CCC2CN3C(=O)C(F)CC(C)C)=O)c1 C=CCCCCCC(=O)N1CC(N(C(=O)C(C)CCCC)C)C(C)(C)C1 c1(NC(C=C(CC)C)=O)sccc1C(=O)N(C(C)C(=O)NC1CC1)C CCN=c1ccc(C(=O)N(C)CC2CC(F)CN2C(C2(C(F)(F)F)CC2)=O)c[nH]1 C(CCCCC)N(CC(=O)N(C(C)CNC(=O)CCc1conc1C)CC)C.CCO C(C(F)C(=O)N1CC(OC2CCN(C(c3ccsc3C(F)F)=O)C2)C1)N(C)CC N1(C(C(CC#C)C2CC2)=O)CCCN(C(c2cnn(C3CC3)c2)=O)CC1C c1(OC)cccc(-c2n[nH]cc2C(c2nnnn2C)NC2C=CCCC2CO)c1 C1(=O)CCC(C)CNC(=O)C2(CC2)CNCC(C)CN1.C1(C)(NC(N)=O)CCC1 N1(C(C=C2CCC(C)CC2)=O)CC(C(N2CC(C(C)O)C2)=O)C(F)(F)C1 c1(N2C(=O)C2)cccc([N+](=O)[O-])c1.Cc1cncnc1-c1cn(CC(Cl)=CCl)nn1 c1(C(=O)NC2C(NC(c3cccc(OCF)n3)=O)C2)cccc(F)c1 N1(C(C2CCC(CC)O2)=O)CCCC(CNC(c2ccc(N(C)C)nc2)=O)C1 C1(C(N2CC(CCCNC(c3n(C)ccn3)=O)OCC2)=O)CC2(CCC2)CCO1 C1(CNC(c2ccnn2C2CCC2)=O)CN(C(C2(C(F)(F)F)CCC2)=O)CCO1 c1(CC)nc2c(C(=O)NC3CC3CNC(=O)CCc3ccsc3)ccnc2[nH]1 O=C1OCc2cc(C(=O)NC3CC4CC3N(C(=O)C(F)=CCCF)C4)ccc21 c1(OC)ccc(C(N2CC(NC(=O)C(F)(F)CC3CC3)C(O)C2)=O)cc1N CC(CC(=O)N=c1cc[nH]c2ccc(I)cc12)C1CCCCC1.C1(=O)CN1 N1(C(C=CCOC)=O)CCC(O)C1.C(=O)(C(C)(Cl)Cl)N N1(C(c2cncc(C)c2)=O)CCC(CNC(C2COCCO2)=O)C(O)C1 C1(C(=O)OCC)(C(=O)NC(CO)C(C)Nc2sccc2COCC)CCCCO1 c1(CC(=O)NCC(CNC(C2CC(F)(F)C2)=O)OC)nc([N+](=O)[O-])n[nH]1 C1(C(=O)NCC2CC(C(=O)NCC3(C(C)C)CCC3)C2)CCCN1C=O N1(C(CCc2cnc(C)nc2O)=O)CCC(N(C(=O)C(C)O)C)C2(CC2)C1 c1(CC(N2CCOC(CNCc3nc(C4CC4)cs3)C2)C)cccc(F)c1 c1(C(=O)NCC2CN(C(CCC#C)=O)C2)ccc(Br)c(O)n1 N1(C(C2(CF)CN(C(C3C(C)CCC3)=O)C2)=O)CC(CO)C1(C)C C(=O)(CCCCCN(C)C)NCC(C1CCOC1)NC(C1CC(C(=O)OC)C1)=O N1(C(=O)Cn2cccnc2=O)CC2CN(C(c3cnc(Cl)[nH]3)=O)CCC2(CO)C1 N1(C(CCC(C)OC)=O)CCN(C(C2CC2C)=O)CC(C)(F)C1 c1(C(N2CCC(NC(C(F)=CCC)=O)C2)=O)oc(SC)cc1C c1(C(N2CCC(N(C)C(c3ccc(O)c(F)c3)=O)C2)=O)cn2ccc(Cl)cc2n1 N1(C(Cc2c(C)nccc2)=O)CC(C(=O)NC2CCN(C)C2(C)C)CC(C)(C)C1 CCCC(C)CC(=O)NC(CCOCCO)C(=O)NCc1cnc(C)cn1 N1(C(CC2(C=C)CN(C(C34CCCN(CC3)C4)=O)C2)=O)CCC(N=[N+]=[N-])CC1 CC1(C)CC(CNC(C2CCCCC2C2CC2)=O)CN(C(=O)CCS(N)(=O)=O)C1 c1(OCCCC)ccccc1C(N1CCCCC1CCCCO)=O C(C(C)CC(=O)NCCN1CCC(NC(c2ccc(OC)nc2)=O)CC1)OC c1(CNC(=O)NC(CC)Cc2cnn(C)c2)c(C)oc2ncnn12 c1(C(N2CCC(C)C(NC(=O)CCC3CCCCO3)C2)=O)n[nH]c2c1CCOC2 c1(OCC)cc(Cl)c(Cl)cc1C(N1CCC1(C)C(=O)NCC1(C)OCCO1)=O C1(OC)CN(C(c2cc(C(C)=O)c[nH]2)=O)CC1NC(=O)CNC=O C1(NCC2(C)N(C(=O)OC(C)(C)C)CCC2)COCC(C)(C)C1 c1(C(N2C(Cn3cc(-c4cc(=N)[nH]cc4)nn3)CCC2)=O)ccc(Cl)c(F)c1 c1(C2c3nnnn3CCNC(C)C(C)N2)ccc(C)cc1.c1(SC)ccncc1 c1(C(=O)NC2CN(C(=O)C(O)CC3CC3)CC2n2ccnn2)cccc(F)c1F C12(C(=O)NCCP(C)(C)=O)CCOC1CN(C(=O)OC(C)(C)C)C2 CC1(CO)CCN(C(C2CCC(NC(c3c(O)ccc(F)c3F)=O)C2)=O)CC1O c1(C(=O)NCC(c2ccc(OCC)cc2)O)cccc2oc(=N)[nH]c12 c1(CNc2cnns2)ccc(CS(C)(=O)=O)cc1.C12(CCC1)N(C(C)=O)C2 c1(CC(=O)NCC(CNC(Cn2c(C)ccn2)=O)(C)C)cccc(C(F)F)c1 N12C(CC1C)C2=O.C1(NC(C2C(COC)CC2)=O)C(C(=O)OC)C1(C)C N1(C(c2cnns2)=O)CCCC2(CCN(c3nc(Cl)nc4c3SCC4)C2)C1 Cc1cc(NC(=O)CNC(=O)NC2CCC(=O)N(c3ccccc3)C2)cc(C)c1 CCC(C)(C)C(C)NC(=O)COCCNC(C1CN(C(C)=O)C1)=O C1(NC(C(CC)C)=O)CCOCC1NC(c1cccc(CN2CCOC2=O)c1)=O C1(C)(C(N(C)CC2N(C(C=CC)=O)CC(F)C2)=O)CCCCNC1=O C1(CNC(c2c(C)ocn2)=O)CCCCN1C(=O)Cn1cccc1 N1(C(C(C)OCCOCC)=O)CC2CCCC(N(C(=O)C(C)(C)CO)C)C2C1 C1(CC#N)CN(C(c2c(O)cccc2Br)=O)CCN1C(c1ccc(Br)cc1F)=O c1(NC(c2c(CC)nco2)=O)ccc(NC(=O)CC23CCC(C)(C2)OC3)cc1C C(C)(C)(CCCNC(C1C(CC(=O)Nc2c(Cl)cnn2C)C1(C)C)=O)OCC c1(C(=O)NCC(CC)NC(c2cc(C3CC3)ccn2)=O)ccc(C)c(F)c1 C1(N(C)C(C2CC3(C2)CC(C)(C)C3)=O)CCOC2(CCN(c3ncccn3)CC2)C1 C1(NC(c2scc(OC)c2)=O)CN(C(C2CCC(C)(C)CO2)=O)CC12CCOCC2 CCCC(C)(O)C(=O)NCC1CCCN(C(c2oc(Cl)cc2C)=O)C1 c1(Cn2cc(CC3N(C(C(C)CF)=O)CCOC3)nn2)ccc(Cl)c(F)c1 c1(OC)ccc(CNc2ccc(NCc3ncccn3)nc2)c([N+](=O)[O-])c1 c1(NCCCC(N2CCC(NC(C=C(CC)C)=O)C2)=O)cccc(C#N)c1 N1(C(c2c(CC)ocn2)=O)CC2CCC2(CCNC(=O)Cc2nccn2C)C1 C=C(Br)CC(C)(C)C(=O)NCC1(NC(C2C(F)(F)C23CCC3)=O)CC1 c1(N2CC(CC)C(O)CC2)nc(N2CCC(C(N)=O)C2)c2ncccc2n1 N1(C(COCCOCCOC)=O)CC2CC1CN(C(c1cncc(SC)c1)=O)C2 C1(CC(=O)NCC(C(C)C)NC(c2n(C(C)C)ncc2)=O)CC(C)(C)OC1=O C=CC(C)(C)CC(=O)N(CCC(C)NC(=O)C(c1ccc(Cl)cc1)(C)O)C C1(NC(C2C(C)CN(C(C3CC3C(F)(F)F)=O)C2)=O)C2CCCC1CC2 C(C1CCOC1)=CC(=O)NC1CCN(C(=O)C(O)C2CC2)C1 c1(OC)cc(C(N2CCN(C)C(CNC(c3cccs3)=O)C2)=O)cc(F)n1 c1(C(=O)NCC2(F)CCN(C(CC(C)CN(C)C)=O)C2)cc(F)ccc1F Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCN(C(=O)CC2CCC(=O)N2)C1C N1(c2cc(OCC)nc(C)n2)CCC(N2CCOCC2C(=O)NC)C(C)CC1 CC1CN(C(c2ccc(Br)c(N)c2)=O)CCN1C(=O)CC1(O)CCOC1 S(=O)(=O)(c1cnn(C)c1)NC1CCN(C)C1.N12C3CCC(C3)C1C2=O C1(N(C(C(C)(O)c2ccccc2)=O)CCO)CCCN(C(=O)CCCCO)C1 C(=O)(CCCC(=O)N(C1CCCN(C(c2cc(C)nc(CC)n2)=O)C1)C)OCC Cc1[nH]c(=N)sc1C(=O)NC(C)(CNC(=O)C(C)(C)n1ccnn1)CO c1(OC)cnc(C(N2CCOCC2CCNC(=O)COC2CCOC2)=O)cn1 CC(C)CC(O)C(C)C(=O)N1CC(O)CC1CC(N1CCC12CCCC2)=O c1(C(N2C(CCCN(C3CC3)CC)CCC2)=O)cnn(C2CCCC2)c1C C12(CNC(C3C(C(=O)OCC)CC3)=O)CC1CN(C(=O)C(C)n1ccnn1)C2.CCOC N1(C(C)C)CCCC(CC(=O)NC2CC(CCNC(=O)Cc3csc(=N)[nH]3)C2)C1 c1(C(=O)NC(CC)CC)ccc2c(c1)CN(C(=O)NC1CC(SC)C1)C2 C12(CNC(CC3CN(C(C)=O)C3)=O)CCN(CC1)CC2 CCC(CC(F)F)C(=O)NCC(C1CCCC1)NC(c1ncn(C)c1C)=O n1(CC)nc(C(N2CCC(C(C(C)C)NC(C3CCN3C)=O)CC2)=O)c(C)n1 c1(C(=O)NCC2N(C(C(C(C)C)SCC)=O)CCC2)cc(O)ccc1N N1(C(C(CC=CC)NC(=O)CCOCC(F)F)=O)CCC2CCN(C)CC12 C1(C)(CC)C=C(C(=O)N2CCCC2CN(C(c2ccc(C(C)=O)nn2)=O)CC)C1 c1(NC(N2CCCC(N(C(=O)CCCN3CCCC3)C)C2)=O)cc(N)c(F)cn1 S(=O)(=O)(c1ccc(F)c(C(C)=O)c1)NC(C(C(C)O)OC)=O C1(C)(OC)CN(CC(=O)NC(C2CCN(C(C3(O)CCC3)=O)C2)(C)C)C1 n1(CC(=O)Nc2ccnc(F)c2F)ccc([N+](=O)[O-])n1 C(=O)(N=c1cc(C)n(CCO)[nH]1)C1(CNC(CCCC(C=C)C)=O)CCCO1 N1(C(C(C)OCC)=O)CCN(C(c2c[nH]c(=N)c(C)c2)=O)CC1C1CCCC1 Cc1nc2ccc(C(=O)NC34CC3CN(C(=O)CCc3c[nH]c(=N)[nH]3)C4)cc2s1 N1(C(C2(C(F)(F)F)CC2)=O)CC(O)CC1Cn1cc(-c2ccc(Cl)cc2)nn1 c1(C(c2n(C)nnn2)NCC2(c3ccccc3)CC(C)C2)ccc(S(C)=O)cc1 C=CCC(C(=O)N1CCC1CC(=O)NCc1nccnc1CC)C(C)C Cc1sc(C)c2sc(C(N3CCC(CN(C)C(C4CCNC(=O)C4)=O)C3)=O)cc12 C(=O)(C(C(F)(F)F)C(F)(F)F)NCC=CCNC(CCc1nc(C)c(C)o1)=O Cc1nc2c(o1)CCN(C(=O)C(C(C)O)CC)C2.C(=O)C(C)CO c1(C(N2CCC(N(C(=O)Cn3cnccc3=O)CC)C2)=O)ccc(C)c(F)c1N C(=O)(C(O)CC(C)C)NC12CC(NC(CC(C)C)=O)(C1)C2 Cc1ccc(F)c(C(N2CC3CCN(C(=O)CC(C)(C)C)C3C2)=O)c1Cl C1(C(=O)NC2(CC=C)CN(C(=O)CCCN3CCCC3)C2)CCOC2(CCC2)C1 CC1(C)CCCN(C(c2csnc2Cl)=O)C1CNC(C1CN2CCCN1CC2)=O c1(CCC(=O)NC2(CNC(C3CC34CCCCC4)=O)CC2)coc2ccccc12 c1(CC(CC(=O)NC2CC2O)NC(=O)CCc2cn[nH]c2)ccc([N+](=O)[O-])cc1 C1(NC(C(=O)NC(c2ncc(CN(C)C)s2)C)=O)CNCCC1C CC(C)(CCNC(=O)Cc1cn[nH]c1)NC(=O)CCN1CCOCC1 C(C(C(=O)N(C1CCNCC1)C1CC1)NC(=O)CC1CC2CC1C2)OC c1(C(N(CCCNC(=O)CCC2CC2(Cl)Cl)C)=O)sc([N+](=O)[O-])cc1Cl c1(C(=O)NCC(CC)NC(=O)C(F)C2CC2)ccc(Br)c(C)c1 c1(C(=O)NC(C)CC2CN(C(=O)C(C)(F)C(C)(C)F)C2)nccc2[nH]ccc12 c1(C(N(c2nccc(OC)n2)C2CCNCC2)=O)cnn2cccc(C)c12 c1(NC(C2CCN(CC3N(Cc4ccn(C)c4)CCC3)C2)=O)ccc(F)cc1 c1(C(N2CC(NC(CC(CC)OC)=O)C2)=O)cc2cccc(Cl)c2cn1 c1(C(=O)NC2CCCN(C(c3[nH]cc(C)c3C)=O)C2C)ccn2cncc2c1 c1(C(N2CCC(N(C(C3CCC(C)CC3)=O)C)C2)=O)cnc2c(Cl)cccn12 c1(OC)ccc(Cl)cc1N(C(C)C)Cc1ccc(C(F)(F)F)nn1 N1(N2C(C=O)(CC)CCC2)CC2C3C=CC(C3)C2C1.c1(C(=O)OC)cccc2cncn12 CC1C(C(=O)NCC(F)F)CCCN1C(=O)C(C)c1cc[nH]n1 C(CCCCF)NC(C1N(C(CC2C(CC)C2)=O)CC1)=O N1(C(c2ccc(NC)c(F)c2)=O)CC2=C(C1)CN(C(=O)C1=CCCC1C)C2 C(C)(N=c1cc(NCCF)nc(C(F)(F)F)[nH]1)C1(c2cccc(C)c2C)CC1 O=CN1CCC(c2nnnn2C2COC2)(NC2COC(C3CCC3)C2)CC1 c1(CC(=O)NC(CNC(c2ccc(C)c(C)n2)=O)C)cn2c(C)csc2n1 C(=O)(C1=CCCC(C)(C)C1)NCC1N(C(c2c(CC)cno2)=O)CC(C)(C)OC1 N1(C(c2c(C)cn(C)c2)=O)CCC(CO)(NC(c2cc(Cl)cnc2O)=O)CC1 c1(C(=O)NC(CNC(C(c2ccc(F)cc2)C)=O)C2CC2)csc(=NC2CC2)[nH]1 c1(C(=O)NCC(C)N(C(c2cnnc(O)c2)=O)CC)cnc(O)cc1C C(CC1CC1)(C(=O)NC(c1cccnc1)C1CC1)NC(c1cc[nH]c1)=O C(=O)(C(C)CC(C)(C)C)N1CCC2C(C(=O)NC(c3cccc(O)c3)C)C2C1 C1(O)(COC)CCC(NC(=O)C(=O)Nc2cccc(N3CCCC3=O)c2C)CC1 C#CCCCC(C)C(=O)NC1(CN(C(=O)CCCCN2CCCC2)C)CC1 CCCC(C(=O)Nc1cccc(NC(c2cc(Br)no2)=O)c1)OCC Cc1cncc(F)c1C(=O)NC1CC(CNC(=O)C=Cc2cccc(F)c2)C1 N1(C(C)=O)CCCC1(C)C(=O)NCCC1(C)CCN(C(c2ncc(F)cn2)=O)C1 C(=O)(C(CCC)=CCC)N(C)CC1N(C(COCCC=C)=O)CCC1 N1(C(C(CNC(C2C(C)CCC2)=O)N(C)C)=O)CC(C)C12CCOCC2 CC1CCC(NC(=O)CCC(C)(C)C)CN1C(C1CN(C)CCO1)=O C#Cc1cc(NC(C23CC(NCc4ccc(Cl)c(O)c4)(C2)C3)=O)ccc1C Cc1ncc([N+](=O)[O-])n1CC(=O)NCCCC(C)NC(c1nccc(Cl)c1F)=O Nc1cccc(C(=O)NOOC(C2CN(CC3CCOC3)CC2C(F)F)=O)c1F N1(C(CN(CC(C)(C)C)C)=O)CC(NC(c2cccnc2O)=O)C(F)C1 C(=O)(C1=CCCSC1)NCCCOCCCNC(=O)NC.C1CC(=O)N1 Cc1cccc(F)c1CN1CC(=O)OC(C)C1 C(=O)(C(C)(C)CC(=O)NCCC1CCCCN1C(=O)CCCCN(C)C)OC Cc1ccc(N2CCOCC2)cc1NC(=O)NCCCCCCSc1cccs1 N1(C(=O)NCc2c(C)nc(Br)cc2)CC(C)OC(C)(C(F)F)C1 c1(C(C(C)C)N(C(=O)COC(F)F)Cc2cn[nH]c2)ccccc1 Cc1[nH]nc2cc(C(=O)NC3(C)CCN(C(C4CC5CCCCC45)=O)C3)ccc12 C1(CC(=O)NCC2CC(NC(=O)CC3CCC4CC34)C2)SC2=NCCN2C1=O N1(CCC)CCCC(C(=O)NC2CCCC(NC(=O)Cn3nnnc3C)C2)C1 c1(SCC(N2CC(NC(C3CC34CC4(F)F)=O)C2)=O)ccc(F)cc1 Cc1ccc(C(N2CC3(CC3)CC2SCC(=O)N(C2CC2(C)C)C)=O)nc1C N1(C(CCCC(C)=O)=O)CCCN(C(=O)CCn2cnc([N+](=O)[O-])c2)CC1CO C1(C(=O)NC(CCCNC(c2c(C)nc(CC3CC3)o2)=O)C)CCCCNC1=O C1(CNC(=O)C=CI)COC2(CCN(C(=O)Cn3cc(CO)nn3)CC2)CO1 c1(C(N2C3CC(CNC(C(C)(C)C(N)=O)=O)(OC3)C2)=O)n[nH]c2ccccc12 N1(C(C2C(C3C(C)C3)C2)=O)CCCC(C2CC2NC(C2(C)CCCN(C)C2)=O)C1 C1(CNC(c2c(CC)non2)=O)CC2(CCN(C(=O)CCC(F)F)C2)CO1 CCC(C)(C)CS(=O)(=O)NC(c1ccc(Br)c(F)c1)c1nccn1C N1(C(COCCCC)=O)CCN(C(=O)COCC2CCCOC2)C2COCC12 CC(C)(C(=O)NCCC1(C(=O)NCCc2ncc[nH]2)CCC1)c1cccs1 Cc1ncnc(N2CCC(C)(CNC(c3cccnc3)=O)CC2)c1Br Cn1ncc(CCC(=O)NC2CC(NC(=O)CCC3CCOC3)C2)n1 c1(C(=O)NC(C)CNC(c2cc[nH]n2)=O)cccc2ncnc(O)c12 C1(C(F)F)(CNC(C(C)=C(CC)C)=O)CCN(C(C2CCN2C)=O)C1 Cc1cc(Cl)c(C(=O)NCC(c2cccc(Cl)c2)NC(C2CC(C)C2)=O)cn1 c1(NC(C2N(Cc3ccc(OCOC)cc3)CC(O)C2)=O)ccnc(F)c1Br C1(NS(=O)(=O)CC2CCCC23CC3)CCc2nn(CCO)cc2C1 CN1CCCC1C=CC(N1CCC(CCNC(C2(C#N)CC=CC2)=O)C1)=O C(C(=O)N1CC(O)CCO1)N(CCC)C(c1cnc(C)[nH]c1=N)=O CC(C)(C)C1=NOC(C(N2CCC(CNC(c3ccc(Cl)c(Cl)c3N)=O)C2)=O)C1 S(=O)(=O)(c1cn(C)nc1C)N1CCCC(C(=O)NC(CCC)C(=O)O)CC1 N1(C(c2cc(C)oc2)=O)CC(C(=O)NC(=O)CCCNc2ccccc2)CC1C Cc1cnn(C)c1C(=O)NCCCN(C(=O)C=CC1CCCN1C)CCO c1(CCN(CC)CC)ccc(N(C(C(=O)NC(C)C)c2cnsc2)C)cc1 C1(CC)CC(C(=O)NCC(C)N(C(c2ccc(NC=O)cc2)=O)CC)CC(=O)N1 N1(C(c2c(C)nns2)=O)CC2CCCC2(C(=O)NCC(C)(C)N2CCCC2)C1 N1(C(C(C)COC(c2ccns2)=O)=O)CCN(C2CC2CNC(=O)COCO)CC1.O(C)C CCC(CC)(CO)C(=O)NCC(=O)NCC1CN2CCC1CC2 CCC(CC)CCCC(=O)NC1CN(C(=O)CCc2cccs2)CC1SC N1(C(CC#N)=O)CCC(O)CC(NC(=O)CCc2nnc(C3CC3)o2)C1 c1(C(N2CCCN(C(CC=C)=O)C(C)C2)=O)oc(P(C)(C)=O)cc1C N1(C(C2=C(CC)OCCC2)=O)CC=C(C(C)(C)C(=O)NCC(CO)OC)C1 c1(CCC(=O)N(C(C(CO)NC(C2C(C(=O)OC)C2)=O)C)CC)ccc(O)nn1 C(=O)(C1=CSCCO1)N(C1CCN(C(=O)C2=NOCC2)C1)C Cc1ccc(C(C)(C)NC(=O)NCCCNc2ncsc2NC2CC2)cn1 C1(CNC(C=CC(=O)N(C)C)=O)(NC(=O)CC2NC(=O)NC2=O)CCOCC1 C=CC(C)(C)CC(=O)NC12CCC(CC1NC(c1cc(C(C)=O)c[nH]1)=O)C2 Cc1ncc(CCC(N2CC3CC2CN3C(C2CC(=O)NC(=O)N2)=O)=O)c(O)n1 C(=O)(C1CCN(C)c2ccccc21)N(CC(CC)NC(c1cccc(O)n1)=O)C Cc1ccn2cc(C(=O)NC3CC4(C3)CN(C(=O)CC(C)C(F)F)C4)nc2c1 c1(C(N2C3CN(C(c4cccc(C#C)c4)=O)C(C3)C2)=O)c[nH]c2ccncc12 N1(C(c2cc(C)nc(O)n2)=O)CCN2C(=O)C(NC(=O)CC3CCCC3)CC2C1 C1(CNC(C2CC(=C)C2)=O)COC(CNC(c2nccn2C)=O)C1 c1(N2CCC(NC(C(C)S(C)(=O)=O)=O)C(C)C2)cc(C#N)ccc1[N+](=O)[O-] C=CC(C)CC(=O)NC1CCC1NC(=O)Cc1nc(C2CC2)cs1 C1(CNC(C2(C#C)CCC2)=O)CN(C(c2ccnc(OC(F)F)c2)=O)CC1O C#Cc1cc(C(=O)NCCC2(O)CCCN(C(c3cc(F)cs3)=O)C2)ccc1C c1(C(N2CCC(CC#C)CC2)C(=O)NCC2C3CCCC23)ccc(Cl)c(Cl)c1Cl C1(C(=O)NCCC2CN(C(C(C)N(C)C)=O)C2)CC(O)CN1c1ccncn1 C(=O)(C(O)COC)NC(C)=O.C1(C(=O)SCC)(CCOCCOCCN)CC1 n1(C(CC)C)nc(CS(C)(=O)=O)nc1NC(=O)CCc1cccnc1 O=C(CCCC#Cc1ccccc1)OCC(Cl)=CCl Cc1noc(C(C)C)c1C(N1CCCCC1c1cn(-c2cccc(F)c2)nn1)=O N1(C(C(C(CC)C)OC)C(=O)NCCSC)CC2CCC(C1)C2(F)F C1(C(=O)NCC2(C)CCN(C(=O)C(O)CC3CCCC3)C2)CCC2(CCC2)CO1 c1(OC)ccc(CN2CCCC(C(=O)N(C)CC3CCOCC3)CC2)nc1Br c1(CC(=O)OC)cccc(C(N2CC3CC2CN3Cc2nonc2C)=O)c1C c1(OC(C)(C)C)cccnc1C(=O)NC1CC(NC(=O)Cn2cnnn2)C1 c1(C(=O)NCC2CCCCN(C(CN(C)CC)=O)C2)c(C)nc(CN)nc1C N1(C(c2c(C)nns2)=O)CCC(C(=O)NCCOc2ccccn2)C(O)C1 C1(CNC(CN(C(=O)C(C)C(C)O)C)=O)CN(C(=O)OC(C)(C)C)CCO1 Cc1csc2c(N3CC4CC3CN4C(=O)CC3CCc4nncn4C3)ncnc12 N1(C(C(CC2(C#N)CCC2)O)=O)CCC2(CNC(=O)C2)C1 c1(C(=O)NC2CC3(COC)C2C3)ccc(Cl)c(C)c1 Cc1cc(C(=O)NCC2(O)CCN(C(=O)COC(C)C)CC2)ccc1C1CC1 N1(c2nc(OC)nc(C)c2)CCC(C2CCN(C(c3nn(C)cc3C)=O)CC2)C1 C1(S(N)(=O)=O)(C(N(CC(C)NC(c2cnc(C(C)OC)s2)=O)C)=O)CCCC1 C1(C(=O)NC2(CNC(C(C=CC)O)=O)CCCCC2C)COc2ccccc2O1 N1(C(C2N(C)CCOC2)=O)CCCC2(CCN(C(c3cnc(O)n3C)=O)CC2)C1 c1(C(=O)NCCC(=O)NC)nc2ccc(-c3cncc(OC)c3)cc2cc1C C1(C(C)(F)F)CCN(C(=O)NC2CC2c2ccc(Br)s2)C1 Cc1c(Br)ccc(C(N2CC3(CC(NC(c4cn[nH]c4)=O)C3)C2)=O)c1C CC1C(NC(=O)CC2CCCC(=O)C2)CCN1C(c1cncc(C(N)=O)c1)=O Cc1ccc(C(CNC(c2c(C)ccn2C)=O)NC(=O)CS(C)(=O)=O)cc1 C1(NC(C(CC)C)=O)CC2CC(C1)N(C(=O)CCCN1CCCCC1)C2 CC1CCC(CC(=O)NCc2csc(C(=O)NCC(F)(F)C(C)O)c2)CC1 c1(C(=O)NC(CC)CNC(c2cc(C3(C)COC3)no2)=O)cc(Cl)cn1C Cc1cnc(C(=O)NCCC2CCN(C(=O)CCCC3CCCCC3)C2)nc1 N1(C(C(C(=O)OCC)C2CC2)=O)CCCCC(NC(=O)CSc2nccs2)C1 C(C(CC(C)C)C(=O)N1CCOC(C(N)=O)C1)Nc1c(C#N)nc(C)o1.C1C(=O)O1 c1(N2C3CN(C(c4c(OCC)ccs4)=O)C(C3)C2)cc(C(C)=O)c([N+](=O)[O-])cn1 N1(C(=O)CN2CCCCC2)CC2CCCN(C(C3CN4CCCN3CC4)=O)C2C1 C1(NC(C2CC=CC2)=O)CCC2CCN(C(C3C4CCC5C(C4)CC35)=O)C1C2 N1(C(COC)=O)CC2(NC(=O)C(c3ccc(N(C)C)cc3)=O)CC1C2 c1(OCC)cc(C(=O)NCC2CN(Sc3cscn3)C(C)C2)oc(=O)c1.C1(=O)CN1 CC(C(C)(C)C(=O)N1CC2(CC2)C1)NC(=O)CC1CC1 Cc1nc2c(s1)CC(C(=O)NC1(CNC(=O)COC3CC=CC3)CCOC1)CC2 n1(CC(=O)NCC23N(C(C(CCC)CC)=O)C(CC2)CC3)cc([N+](=O)[O-])c(C)n1 c1(CC)ccc(NC(C2C=CCCN2C(=O)CC2CCOC2(C)C)=O)cn1 C(C(C)(C(=O)N1CC(O)C(O)CO1)NC(c1cc2cccnc2[nH]1)=O)SC c1(NC2C(OC)CCCC2)ccc(Br)c(C)n1 N1(C(CN(C)C)=O)CCC(C)(C)C1CC(=O)NCCN(C)C.C12CN(C1)C(=O)O2 C(=O)(C(C)C(=O)NCCCOCCNC(=O)CNC(=O)C(F)(F)F)OC Cc1cc(Br)c(N)cc1NCC(=O)NC(c1ccnn1C)Cc1ccccc1 CC(C)C(CC1CCCC1)C(=O)N(CC)CC1CCCN(C(=O)C(C)C(C)C)C1 C1(NC(c2nc(C)[nH]n2)=O)CN(C(=O)C(C)CSC(F)(F)F)CC1C(F)(F)F N(C)(C(=NCCC1(C)CC1(F)Cl)NCCNC(C)=O)CCCCOC N1(C(CCCCCOC)=O)CCCN(C(C2CC(N(C)C)C2)=O)C(CO)C1 C1(CC(=O)N(C(=O)CC2CCC2)C(C)C)CCN(C(=O)CC2CC=CC2)C1 CC(C)(C)CC(O)C(=O)N1CC(C2CN(C(=O)CC3CCOCC3)C2)C1 Cc1cncc2cc(C(N3CCC(C(CO)NC(=O)CCC(N)=O)CC3)=O)sc12 c1(C(N2C(C)(CNC(=O)C(O)C3CC3)CCC2)=O)nc(Br)n2ccccc12 C(=O)(C1CCCc2nccn21)N(C)CC1CCCN1C(c1ccoc1)=O c1(C(=O)NC(C(C)NC(c2c(Cl)cc(C)s2)=O)CO)ccn2c1CCCC2 N1(C(CC(CC)OC)=O)CCCC(C2(NC(C3CCC(C)CC3)=O)CC2)C1 C#CCCCCNC(=O)C(c1cn(C)nn1)NC(=O)COC(C)=O CCCCCCC(F)C(=O)N1CC2CCC1CN2C(c1cc(N)cc(F)c1)=O C1(NC(C(C)=CC2CC2)=O)CCCN(C(=O)C(C)Cc2ccccc2C)C1 c1(C(=O)NCCC2CC(NC(c3c(C)oc(C)c3C)=O)C2)cnc2[nH]cnc2c1 c1(C(N2CC(C)C(CNC(c3ccoc3)=O)C2)=O)sccc1S(=O)(=O)C(F)F N1(C(CC2(N(C(c3c(C)cnnc3)=O)C)CC2)=O)CC(F)(F)CCC1C c1(C(CC)C)ccc(CC(=O)NC2(C)CN(C(=O)C=CCn3ccnn3)C2)cc1 c1(C(N2C(CC(=O)Nc3cc(F)ccc3O)CC(O)C2)=O)ncc(F)cc1F C1(NC(c2c(OC)n(C)nc2)=O)CN(C(=O)C(C)(C)C2CC2)CC1(C)C Cc1nnc(O)c(C(=O)NCC2(C)CCN(C(c3ccc(F)cc3Cl)=O)C2)c1C c1(C(N2CC(CC=C)(NC(C3CN(C(N)=O)C3)=O)C2)=O)csc2nccn12 N1(C(C2N(CCCC)CCOC2)=O)CCC(NC(=O)C(C)(Cl)Cl)CC(C)(C)C1 c1(OC)ncnc(C(=O)NC(C2CCCN2C(=O)CCC2CC2(F)F)C)c1F C=C(C)CC(C(=O)NCCOC)NC(=O)CN1C(=O)CCCC1=O N1(C(C2(C)C(CC)CCC2)=O)CC(C2(NC(=O)CC3CCC4(CCC4)O3)CC2)C1 C1(NC(CCOCC#C)=O)CCCC(CNC(=O)C(C)(C)C2CC2)C1 c1(C(=O)NC(c2cnc(C)s2)C)c(CNC(=O)CNC(=O)C(C)(C)C)cnn1C c1(C(N(C)CC2CCCN2C(C2CC3(CCC3O)C2)=O)=O)cc2cccnn2n1 c1(C(N2CC(NC(C3(C(O)C(F)(F)F)CCC3)=O)C3CC23)=O)ccc(CO)cc1 C(=O)(C1=NOC(CNC(C2CC3CCC(C2)O3)=O)C1)NCC1(C)CCOC1 N1(Cc2cn(COC)nn2)Cc2ccc(Br)cc2C1.C1CO1 O=S(=O)(c1cc(F)c(F)c(Cl)c1)NC1CC(F)CN(Cc2cnc(C3CC3)s2)C1 C1(C(=O)Nc2noc(-c3coc(C4CC4)n3)n2)COc2ccc(F)cc2C1 C1(C(C)C)CCC(C(N2CC(C)(F)C2)=O)N1C(c1cnc(N(C)C)cn1)=O c1(NC(C2(CNC(=O)CNC3CC3)CCC2)=O)cccc(N2CCCC(O)C2)c1 CC(CC(=O)N1CCCN(C(c2ccc(F)c(C3(C)CC3)c2)=O)CC1)C(F)(F)F c1(C(N2CC(NC(C(C(C)OC)O)=O)C2)=O)cc(C)cc2c1CCC2 c1(C(=O)NCCCC(C)NC(C(CC(C)C)OC)=O)cc2c(cc1F)NCCC2 n1(CC)cc([N+](=O)[O-])c(=NCC(=O)NCC(C)(C)NC(=O)C=CC(=O)NC(C)C)[nH]1 C1(CNC(C(=O)NC(C)C)=O)CN(C(=O)C(=O)CCc2ccccc2)CCCO1 c1(C(=O)NC2(C)CC(NC(C(C3CCC3)OCC)=O)C2)cc(N)c(F)cn1 C(CCC1CC1)(C(=O)Nc1ccc(OC)nc1)NC(C1CC(O)(CC#C)C1)=O N1(C(Cc2ccn(C)n2)=O)CC(NC(=O)C(F)(F)CO)C(F)C1 Cc1cc(C(=O)NC2CCCC(C(=O)NCc3cnn(C4CC4)c3)C2)ccc1Cl C1(NC(CC2(C=C)CC2)=O)C2CC3CN(C(c4c[nH]nc4OC)=O)C1C3C2 Cc1sc(C)c(C(N2CCC(NC(c3cccnc3)=O)CC2C)=O)c1C c1(C(=O)NC2CCN(C(C(CC)C(=O)OC)=O)C2)cc2cc(F)cc(F)c2[nH]1 CN1CCC(C(=O)NC2CC23CC(NC(=O)CCC2(C)CC2)C3)CC1 CCC(C)CCC(O)CC(=O)NC1CCC(CNC(C2CCC=CCC2)=O)C1 N1(C(c2cnn[nH]2)=O)CCOC2(CCC(N=c3ncc4ccccc4[nH]3)CC2)C1 c1(C(=O)NCC2CC(NC(CCC)=O)C(O)C2)nc2ccccc2[nH]1 C(=O)(CCCCCNC(=O)COc1ccn(C)n1)N1CCN(C)CC1 c1(N2CC(C)=C(C)CC2)[nH]c(=NCCN2C(=O)CCC2=O)nc2sccc12 Cc1cc(C(C)(C)C(=O)NC2(CCNc3nc(C4CC4)ns3)CCCC2)cs1 C1(n2cc(-c3cnc(OC)s3)nn2)CN(C(C2CC2(C)C(=O)O)=O)CC1O Cc1ncc(C(N2CC(C(=O)NCC(N3CCOCC3)=O)C(F)C2)=O)c(C)n1 c1(C(=O)NC2CC(CNC(=O)Cc3cncnc3)C2)cccc2sncc12 N1(C(c2c(C)cncc2)=O)CC(NC(C2CSCC(=O)N2)=O)CC(C)C1 c1(C(=O)NCCC2OCCN(C(C3C(C)(CC)C3)=O)C2)cc2sccc2[nH]1 CC1CN(C(=O)C(=O)Nc2ncc(-c3ccccc3)s2)CC(C)(C)O1 C=CCC(CC(=O)N1CCOC(C)C1CO)NC(=O)CCCSCC C1(CCNC(C2CC(C)(CC)C2)=O)CC2CCC(C1)N2C(=O)C(C)NS(C)(=O)=O N1(C(c2cn(CC(=O)N(C)C)nn2)=O)CCC(NC(=O)C(COC)N(C)C)CC1 c1(C(=O)NC(CC)CNC(=O)C(C2CCOCC2)F)cc(Br)ccc1OC c1(C(=O)NC(CCCNC(c2n(CCC)ncc2)=O)C)ccc(Cl)c(C)c1N C1(SCc2nc(C)on2)CCC2C(CC1)C2(F)F.N12CCC(CC1)C2 C1(NC(c2ncc(N)nc2)=O)(CO)CCCN(C(=O)Cc2cnccn2)C1 CCCCC(C(=O)N1CC(C2(OCC(N3CCCC3)=O)CC2)C1)OC.C1(=O)CN1 C1(OCC)CCCN(c2nnc(C(C)NS(C)(=O)=O)n2CCc2nc(C)c(C)s2)C1 c1(CCCc2scc(C)n2)nc(Cn2cccn2)nn1-c1ccnc(Br)c1 N1(C(C2(C#C)CN(C(=O)C(C)OCCOC)C2)=O)CCCC(O)(CC)C1 N1(C(C2C(CNC(C3(COC)CCC3)=O)C2(C)C)=O)Cc2cccnc2C1 Cc1ccccc1OCCC(=O)NCC1CCCN1C(c1cocn1)=O c1(CN2CCC(c3n(C(CC)C)nnn3)(OC)CC2)c(OC)ccc(F)c1C c1(C(=O)NC(CNC(c2c(C)[nH]nc2C(C)C)=O)C(C)(C)C)cc(Cl)cc(Cl)c1 c1(OC)ccccc1C1CCN(Cc2ncc(-c3cc(C)nn3C)cn2)CC1 c1(NC(C)CN2CCCNC2=O)c(C)cccc1C C1(C)(CC)C=C(C(=O)NC(C2CCCCC2)C(=O)NCCC#CC(C)(C)C)C1 C=CCCCC(=O)NCc1ncoc1CCNC(c1coc(C)c1)=O C=CC(C)(C)CC(=O)N1CCN(C(=O)COc2cc(F)cc(F)c2)CC1C Cc1ccc2c(c1)C(N(C(=O)Nc1cc(C(=O)O)c(Cl)cc1Br)C1CC1)CCCO2 N1(C(c2c(C)ccc(O)c2)=O)CCC2CN(C(c3ccc(Br)cc3Br)=O)CC12 c1(C(=O)NC2CCC(CCNC(C(CC)N(C)C)=O)C2)cc2c(nn1)CCOC2 c1(C(C(=O)OC)NC(=O)NCC2(C)CCC2)ccc(OC)c(Cl)c1 N1(C(C(CC#C)CC#C)=O)CCC2(CCN(C(=O)C=C(C)CCCC)C2)C1 C1(NC(CC2(C)CCCO2)=O)CCOCC1NC(c1coc(Cl)c1)=O O=S(=O)(c1ccc(Cl)cc1Cl)N1CC2CC(CN(Cc3cc4sccn4c3)C2)C1 C1(C(CNC(=O)C=C2CCCC2)NC(c2ncoc2Br)=O)CCCCC1 C1(CNC(=O)C(O)C2CC2)CN(C(C2CCC=CCC2)=O)C2(CCOCC2)C1 C1(NC(c2ccc(CCCC)cc2)=O)(CC)CCCN(C(=O)CN2CCC2C)C1 C=CCC(C)(C)CC(=O)NC1C=CCCC1C(=O)NCC1CC2(CCO1)CC2 C1(CNC(c2c(NC)c(F)ccc2)=O)CN(C(=O)C2=C(Cl)CC2)CCC1(C)C c1(NCC(CCCC)NC(C(C)=CC)=O)ccc(F)c2occc12 c1(CC(=O)N(C2CCN(C(C(C)(C)SC)=O)C2)C)oc2ccccc2c1C C1(CNC(c2nc(C)oc2)=O)CC2(CCN(C(=O)CCC=CBr)C2)CO1 N1(C(c2c(CC)ccc(F)c2)=O)CC2CC1CN(C(=O)CS(=O)(=O)C1CC1)C2 N1(C(C23CC(C)(C2)C3)=O)CCCC(N(C(=O)CSc2ccccc2O)CCF)C1 c1(C(=O)NC(C2CCN(C(c3cnn(C)n3)=O)C2)C)c(F)ccc(Cl)c1N C(=O)(C(C)(C)CC(=O)N1CCC(CF)(NC(=O)C(O)CN(C)C)C1)OCC C(=O)(C1=CCCN(C(=O)CC2CCC(C#N)C2)C1)N1C(C(C)(C)N(C)C)CCC1 C1(C(=O)NC(CN(C)C(C2(O)COC2)=O)(C)C)COC(=O)C1 c1(COC)nc(C(=O)NCC(C(C)C)NC(c2conc2C2CCC2)=O)co1 n1(Cc2c(C)cccc2)cnc2ccccc2c1=O.c12nc(no1)SCCC2 C1(CC(=O)NC2CCN(C(C(C)=CC3CC3)=O)C2C)CC2CCC1O2 Cc1cc([N+](=O)[O-])cc(C(=O)NC2CC(NC(C3CCC=CCCC3)=O)C2)c1Cl N1(C(C)=O)CC(O)CC1C(=O)N(C)CCNC(=O)C=Cc1ccn(C)c1 N1(C(C(C)(CO)NC(=O)CCC(N)=O)=O)CCC(C2CCCC2)C1 N1(C(C(C2CCCC2)NC(c2cnc(C)o2)=O)=O)CC2(CCNC2=O)C1 C#CCCCC(C)(N)C(=O)N1CCC(C(=O)N(O)CCC(F)(F)F)CC1 CCCC(C(F)(F)F)NC(C1(CCNC(=O)CN2CC(C)(C)C2)CC1)=O CS(=O)(=NC(=O)C1(S(=O)(=O)C2CCCCC2)CC1)c1ccccc1Cl C1(C(=O)NCCn2cc(CN)nn2)CC(=O)N(C)C1.CC1CC1(F)C(=O)C1CC1 N1(C(C2N(C)CCCC2)=O)CC2C=CCC(C2)C1 N1(CC(C)C(N(C(C)C)C)=O)CCN(C(=O)CC2CC3(CCC3)C2)CC1 c1(C(=O)NCC2(C)CCC(NC(c3cc(Cl)no3)=O)C2)ccc(O)nc1Cl c1(C(=O)OC)cc(OC(C)(C)C)c2ncccc2c1.N12CCC(C1)OCC2=O c1(NC(C)=O)ccc(C(=O)NC2CN(C(=O)COCCO)CCC2C)cc1F c1(OC)ccc(C(=O)N(C)CC2CCCN2C(c2nn(C)c(C)c2Cl)=O)cc1O Cc1cc([N+](=O)[O-])cnc1C(N1CCCC(CO)(NC(=O)CSCC#N)C1)=O Cc1ccc2c(c1)c(CNC(=O)NC1CCCC1(C)C)cn2CCNC1CC1 N1(C(c2c(C)n(C)cn2)=O)CC2(CC2)CC1C(=O)NCCCc1ccon1 C1(NC(c2cn(CCO)nn2)=O)CC(=O)N(C2CN(C(c3cnc[nH]3)=O)C2)C1 c1(C(N2CC(CNC(CC(C)(C)c3ccccc3)=O)OCC2)=O)cc(Cl)cc(I)c1 c1(C(=O)NC(C)(C)CNC(=O)Cc2cccc(Br)c2)ccc(N)c(Cl)n1 c1(C(=O)NCCCNC(c2c(C(C)C)ncs2)=O)cnccc1C(F)(F)F n1(CCOC)cc(-c2cn(CC(=O)NC(C)C(C)SC)nn2)cn1 N1(C(c2scc(OC)c2)=O)CCC2CCC(C1)N2C(C1(C)CC=C(C)CC1)=O C=CCCC(C(=O)NCCC1(CO)CC1)NC(C1CC(N(C)C)C1)=O Cc1cc(C(=O)NCCOC(C)C)ccc1-c1cn(C2CCC(=O)N(C)C2)nn1 c1(N2CC(C(=O)Nc3cc(C(=O)OC)c(Cl)nc3)C2)nc(Cl)c2c(n1)COC2 N1(C(CC=C)=O)CCCC1(C)CCC(=O)NCCCC1CCCCO1 Cc1ccc(Cl)cc1OCC(N1CCC1CNC(=O)CC1CCNC1=O)=O CN1CCC(C(=O)Nc2ccc(O)cc2)(NC(=O)CC2CC3CCC2C3)C1 c1(C(=O)NCC(C2CC2)NC(C2(CCC=C)CCCC2)=O)cnn(C2CC2)c1F C(c1ccc(F)c(F)c1)=CC(=O)N(CC(C(C)C)CO)C1CCN(C(C)C)C1=O c1(-c2c(C(=O)NCCCNC(c3ccc(F)s3)=O)nco2)ccccc1F CC(CC(C)(C)C)C(=O)NC1CC1CNC(c1[nH]cc2c1CCCC2)=O Cc1ccc(C(N2CC3C(C(=O)NCCc4ccc(F)cc4)C3C2)=O)cc1C c1(CCC(N2CC(NC(CCOCC(C)C)=O)(CF)C2)=O)ccc(F)cc1 N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CC(NC(=O)CC(C)C)CC12CCCCC2 Cc1c(C(=O)NC2CC(NC(c3cc(F)cc(F)c3)=O)C2)ccc2c1OCCO2 C1(C(=O)NCCOCCNC(=O)CC2CCC3CC23)CC(=O)N(O)C1 N1(C(C(=O)Nc2c(C)cccc2)=O)CCCN(c2ccnc(Cl)c2)CC1 c1(OCC)ccc(F)c(C(=O)NCC(O)CNC(C2(C)CCCC2)=O)c1N c1(SCC(N2C3(CNC(CSCC#C)=O)CC(C2)C3)=O)nc2ccccc2[nH]1 C#CCC(CC(F)F)NC(=O)C=CC(C)(C)NC(=O)CCN(C)C C(=O)(C1=NNC(=O)CC1)N1C(C)CC(NC(c2cc(C)c(O)cc2)=O)C1 CCC(CC)(CCC(=O)NC1CC(F)(CNC(c2c[nH]c(=NC)s2)=O)C1)[N+](=O)[O-] Cc1nn(C)cc1CC(N1CCN(CC(N2CC(C)(F)C2)=O)CC1)=O c12ncc(F)c(n1)O2.N1(C(COCc2onc(CC)n2)=O)CCN(C(C)=O)CC1 c1(CNC(C2CC(C)CC(C)C2)=O)cccc2cn(C)nc12 c1(C(=O)NCCC)ccc(-c2cc(C(=O)N(C)CCN(C)C)ccc2C)c(F)c1 N=c1c(C(N2CCCN(C(=O)Cc3cc[nH]n3)CC2)=O)c[nH]c2ccccc12 C12(C(N3CCC(CC#N)C3)=O)CC(CN1C(=O)Nc1ccc(Br)cc1)C2 N1(C(c2nnn(C)n2)=O)CC2(C)CN(C(c3ccc(=N)[nH]c3)=O)CC2(C)C1 c1(CCNC(=NCCC#C)NCC2COC(C)C2)c(C)[nH]c2ccccc12 C1CC(C(=O)NC)N1.C(C)(C(N)=O)N(C(C=[SH]C)=O)CCC.C(C)(=O)OC c1(C(=O)NCC(=O)NC2CC2NC(CCC(C)C)=O)ccc2c(c1)CCC(=O)C2 N1(C(C(CCC)NC(c2cnc3n2CCC3)=O)=O)CC(C)(C)OCC1C N1(C(CCC=C)=O)CCC(C)C(NC(=O)Cn2cc(C3CC3)cn2)C1 c1(CCC(=O)NC(c2cccc(Cl)c2)CNC(CC=CCC)=O)cccc(F)c1 c1(NC2CCN(C(C(=O)N(C)C)=O)C2)cnc(Cl)c(Cl)c1 C1(COCC)CN(C(C2(C(=O)NCC3CC3)CCC2)=O)C1.C1(C(=O)OC)CC1 c1(C(=O)NCCN(C(CC(C)CN(C)C)=O)C)ccc(Br)cc1O C(=O)(C1=CCC(F)(F)CC1)NC(C1CN(C(c2cc(C)cc(O)n2)=O)C1)C c1(CCC(C)NC(=O)NC2CCCN(CC)C2)cc(OC)cc(OC)c1 Cc1nn(C)c(Cl)c1C(=O)N(C1CCC(NC(C2CCCCCC2)=O)CC1)C N1(C(c2cc(C)cc(C)c2)=O)CC2CCC1CN2C(C1CC(=O)N(C)C(=O)N1)=O c1(C(N2CCC(Oc3cc(C(=O)OC)ncc3)CC2)=O)ccc(S(C)(=O)=O)cn1 C1(NC(C(c2n(C)ncc2)O)=O)CCC2CN(C3CCC=CCC3)CC2C1 Cn1ccc(C=CC(=O)NC2CNCC23CC3)c1 Cc1ccc(Cl)c(NC(=O)NC2CC2C(=O)NCc2cccc(F)c2C)c1 c1(OC)cc(C)c(C(=O)NC(C2CCN(C(C3(C)CCCC3)=O)C2)C)cn1 C12(NC(CCOCCOC)=O)CCOCC1CN(C(=O)C(C)SC(C)C)C2 Cc1c[nH]cc(C(=O)NC2COCC2NC(c2ccc(Cl)c(F)c2)=O)c1=O c1(C(=O)OCC)ccnc(CNC2CCN(C(=O)C(O)CC3CCCC3)C2)c1 c1(C(=O)NC(CCCNC(c2c(CC)n[nH]c2)=O)(C)C)cnc2n1CCOC2 c1(C(N(C(c2c(Cl)cccc2Cl)C)C)=O)cc2c(s1)CCCCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NCC1C2CCCCC12)C1(C)CC1 N1(C(CCC(=C)C)=O)CCN(C(=O)CC2CCCNC(=O)C2)C2CCCC12 c1(NC(C)C)ccc(Cl)c(CN2CCC(CC(=O)Nc3nccs3)CC2)c1 C1(C(C)N(C)C)CCCCN1C(=O)OC(C)(C)C.C12C=CCN(C1)C2=O C1(NC(c2cc(OC)ns2)=O)CC2CCCC(C1)N2C(C1(F)CCN(C)CC1)=O C1(C(N2C(F)(CNC(C(C(C)(C)C)NC(=O)OC)=O)CC2)=O)CCn2nccc2C1 c1(C(N(CCN(C(C2(C)CCC(C)C2)=O)C)C)=O)csc(=NC2CCCCC2)[nH]1 c1(C(N2CC3CN(C(c4scc(C)c4)=O)C3C2)=O)ccc(C#N)cc1I C(CC(C)C(C)(C)C)C(N1CCC(C)C1C(=O)NOc1ccccc1F)=O C(CNC(=O)CC1CCN1C(CC)CC)(C(C)C)NC(C=CCN(CC)CC)=O N1(C(Cc2cnc(C)s2)=O)CCC(CNC(C2CCCC(O)C2)=O)C12CC2 C1(C(=O)NCC2(CNC(c3c(CC)[nH]cc3)=O)CC2(F)F)CC2CCC(C1)N2C Cc1cncc(C(N2CCN(CCNc3ncc(C(F)F)cn3)CC2)=O)c1 CC1(C)CCC(CC(=O)NCc2n[nH]cc2C(=O)NCCN=S(C)(C)=O)O1 C1(NC(C(CCN(C)C)NC(=O)CCCn2cccn2)=O)CC2CC3C(C2)C13 Cc1noc(CNC(=O)NC(COC(C)(C)C)C(F)(F)F)c1C CC1(C)CCCCC1C(N1CC(NC(C2CC(Cc3ccccc3)=NO2)=O)C1)=O C12(C(=O)NC(C3CCCN3C(=O)CSCC3CCCO3)C)CC(C)(C1)OC21CCC1 C(=O)(C1=CCCOCC1)NCCN(CCOC)C(c1[nH]c(C2CC2)nc1C)=O C1(CNC(CNC(C)=O)=O)CCCC1C(=O)NCCNC(N)=O CCCC(C(=O)N1CCC1C)NC(=O)C(C1CC1)OCC.C(C)(C)OC n1(CC(=O)NC2CCC(F)(CNC(c3cc(C)nn3C)=O)C2)cc(F)ccc1=O C(C(CNC(C12CCCC1(C(N)=O)C2)=O)C(F)(F)F)NC(Cn1c(C)ccn1)=O c1(C(=O)NCC23C(CN(C(Cn4ncn(C)c4=O)=O)C2)C3)cnn2cccc2c1 c1(CC)ccc(C(=O)NC(CO)CCCNC(=O)C2CC2)cn1 c1(NC(CN(C(C(C(CC)(C)C)O)=O)C)C)ncc(C)c(S(C)(=O)=O)n1 c1(CC)cnsc1C(=O)NC1(C)CC(NC(C2(O)CC(CF)C2)=O)C1 C1(OC)CN(C(=O)C(c2cnn(C)c2)NC(=O)C(C)n2ccnn2)C2(CCC2)C1 C1(C(N(C(C2CCC2)C)CC)=O)CCC(NC(=O)CCc2cncs2)C1 c1(C(N(C2CCN(C(=O)C=Cc3ccoc3)C2)C)=O)cc(OCC2CC2)ccn1 c1(NC(=O)NCC2(c3ccccc3)CC2(F)F)cnn(-c2ccccc2)c1 c1(C(N2C(C(=O)NCC3CC(COC)C3)CCC(O)C2)=O)cccn2ccnc12 Cc1cc(C(=O)NCCNC(C2CCN(C)C2)=O)oc1C c1(C(N2CC(N(S(CC)(=O)=O)C)C2)=O)cnoc1-c1ccc(Cl)s1 c1(C(=O)NC(CCNC(C2(OC(C)C)CCC2)=O)C)cc(C2CC2)ns1 N1(C(c2nc(CCCCC)sc2)=O)CCN(C(c2csc(C)c2N)=O)CC1CO c1(OC(C)C)ccc(C(=O)NCC(C)(O)CNC(C2CCC(CO)O2)=O)cc1 C1(C(N(C)CCn2cccn2)=O)C(C2CC2)CCN1C(=O)C=Cc1ccc[nH]1 c1(C(=O)OC)c(CNC(c2nnnn2C(C)(C)C)c2cnoc2)ccn1C N1(C(c2[nH]cc(C(C)=O)c2)=O)CC2(C=C(C(=O)N3CCC(O)C3(C)C)CO2)C1 C=CCC(CNC(C1CC=CC1)=O)C(=O)NCC(N)=O c1(C(=O)NC2CCCN(C(C3OCCN(C)C3=O)=O)C2)cnn2c(=O)cc[nH]c12 c1(NC(c2cc(Cl)ccc2Cl)c2n(C(CC)(C)C)nnn2)cc(F)c(O)cc1C CC1=C(C(=O)NCC2(Nc3ncnc4c3nnn4C)COC2)S(=O)(=O)CCO1 C1(NC(C=C(C)C(C)C)=O)CC(N=c2ccnc(C(C)C)[nH]2)C12CCC2 C1(NC(C(CC)CC)=O)CN(C(c2c(Cl)n[nH]c2C)=O)CC1C1CC1 c1(C(C(=O)N(CC(CN(C(CSC(C)C)=O)C)O)C)C)ccc(F)cc1F C1(C)(C(=O)NCC2CCN(C(c3n(C)[nH]c(=N)c3)=O)C2)CC2CCC1O2 N1(C(COCCCC)=O)CC(F)CC1CN(C(=O)CS(=O)(=O)N(CC)CC)C C1(NC(c2nc(COC)sc2)=O)CN(C(=O)C(C)CN(C)C)CC1(C)C c1(OC)cc(NC(=O)C(N2CCC(O)(CC#N)C2)=O)ccc1C c1(C(C)(F)F)ccc(NC2CC3CC2CC3=O)cc1F c1(C(N2CCC(O)CC2)C(=O)NCCCSC)nc(C2CC2)n(C)n1 C(C(O)CC(=O)NCC(C)N(C)C)NC(c1ccc(CNC(C)=O)o1)=O c1(C(=O)NC(CN(C(c2n(CCOC)ncc2)=O)C)C)cccc2c1C(=O)CC2 c1(C(C(=O)NC(C)CCNC(=O)Cc2ccon2)N(C)C)ccccc1F C(C(O)CC(=O)NC1CC(CO)C2CC12)NC(=O)COCC1CC1 c1(C(N2CC(C(C(=O)OC)OC)C2)=O)sc(OC2CC2)nc1-c1ccccc1 c1(OC(c2ccc(F)cc2)C(=O)OC)ccc(Br)c(C)c1I c1(OC)ncc(F)cc1C(N1CCCC(C(=O)NCc2ccccc2C#N)C1)=O Cc1ncccc1C(N1CC(=O)CC1C(=O)N(C)C(C)C1CC1)=O N1(C(c2c(C)ccnn2)=O)CC(O)CCC1C(=O)NC1CCOCC1C C1(C)(CC)CC(NC(=O)C(F)=C(C)C2CC2)CN1C(=O)Cc1ccc(F)cc1F c1(NC(C2CC(O)CN(CC(F)F)C2)=O)ccc(N2CCOCC2)c(Cl)c1 c1(C(=O)NC2C(C)N(C(=O)CNS(=O)(=O)N(C)C)CCC2)cn2c(n1)CCCC2 N1(C(c2onc(OC)c2Br)=O)CC(NC(=O)CN2CC(C)(C)C2)CCC1C c1(CC)cc(C(N2CCCC(NC(c3nccnc3N)=O)CC2)=O)cc(O)n1 c1(C(=O)NCCN(C(c2sccc2C(C)(C)C)=O)CC)ncccc1Br C1(C(N2CC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C(F)C2)=O)CCC2(CC1)CC2 c1(C(C)(C)C)ccc(CNC2(C(F)(F)F)CCOC2)c(O)c1 c1(CC)ccc(C)c(C(=O)N(CC)CC2CCN(C(=O)CS(=O)CC)C2)c1 c1(OC)cc(F)cc(C(=O)NCC2CCCCN2C(=O)C(C)(C)OC)c1N N1(C(c2n(CC)ccc2)=O)CCCC(NC(=O)CCCCOC)C1C C1(C2(NC(C3(C(N(CC4=CCSC4)C)=O)CC3)=O)CC2)CCCCO1 c1(C(N2CC(C(N3CCC(C(=O)OC)C3)=O)OCC2)=O)c(C#N)ncn1C C(=O)(C1=CSCCO1)N(C1CCN(C(=O)CC2CCC(C)(C)CO2)C1)C Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)CCC2CC(C)C2)nn1C(C)C c1(C(CNC(C=CC(=O)NC)=O)NC(=O)CN(C2CC2)CCO)cccc(Cl)c1 N1(C(CCC)=O)CCOC(C)C1C(=O)O.N12CCC(C1)N(CC)C(=O)C2=O C1(C(=O)NCC(C)(C)OCCNC(CC)=O)CCc2cnn(CC)c2C1.C(COC)SCC n1(CC)cccc(NC2(c3nnnn3C(C)COC)CC3CSC3C2)c1=O N1(C(c2ncc(C)cn2)=O)CCC2(CCCC2NC(C2CCSCC2)=O)C1 Cc1cc(Br)ccc1C(=O)NCCC1(NC(C2CC23CCCC3)=O)CC1 C1(C(=O)NCC2CCC(C)CN2C(c2cc(Cl)sc2Cl)=O)CCn2nnnc2C1 N1(C(C(c2ccccc2)OC)=O)CCCC(NC(=O)C(=O)NCC2CC2)C1C O=C(CC=C(Cl)Cl)N(C1(C(=O)NOCCCCC2CC2)CCC1)C1CC1 C1(C(=O)O)CC2(CC(NC(C(n3cc(-c4cnccc4Cl)nn3)C)=O)C2)C1 Cc1cc2c(C(=O)NC3CCCC3NC(=O)CC3(C)CC(F)(F)C3)cccc2[nH]1 C1(c2cn(Cc3c(C)c[nH]n3)nn2)CCCN(C(C2CCCN2C)=O)C1 c1(C(N2CC(C(=O)Nc3cnsc3)C(O)CC2)=O)cc(Br)cc2[nH]ccc12 c1(C(=O)OC(c2ccc(C)s2)C(=O)OC)nn(C(C)C)cc1I N1(C(CCN(CCCCC)C)=O)CCOC(CNC(=O)CC2CC2(Cl)Cl)C1 c1(OC)cc(C(=O)NCC2COCC2NC(C2CCCCS2)=O)ccn1 N1(C(C2C(C3C(C)C3)C2)=O)CC(C2CCCN(C(c3ncccc3F)=O)C2)C1 C(=O)(CC(C)(C)CN(C)C)NC1C=CCC(C(=O)NCC(C(CC)C)O)C1 C1(NC(C2(OC)CCSC2)=O)CN(C(c2cccc(COC)c2)=O)CC1C C=C(Cl)CC(C(=O)N(C)Cc1cnc(C)cn1)NC(c1cnccc1Cl)=O c1(C(C)NC2CCOCC2N2CCOCC2)nc2ccccc2s1 N1(C(C=C(CC)C)=O)CC(CO)C2(CCN(C(=O)C(C)n3cccc3)CC2)C1 N1(C(c2cnc(OC)s2)=O)C2CCC1CN(C(=O)CC1CCOC1)CC2 CC1(CNC(c2c(F)cccc2Cl)=O)CCCN(C(C2(S(N)(=O)=O)CC2)=O)C1 C1(N(C(c2nc(=N)[nH][nH]2)=O)CC)CCCN(C(=O)Cc2cnn(CC)c2)C1 c1(NC2CC(C(=O)Nc3c(CC)cccc3F)C2)ncc2ccc(F)cc2n1 N1(CC2(C3CCCCO3)CC2)c2ccncc2N2CCC1C2 c1(C(=O)NCCC2CN(C(C=CC(C)(C)SC)=O)CC2C)cc(N)nc(Cl)c1 CCCCC(C)(CO)NC(=O)C=CC(C)NC(=O)Cn1ncccc1=O C(=O)(C(C)C(C)NC(C1C=CC(NC(C23CCC(OC)C2C3)=O)C1)=O)OC c1(OCOC)cc(CNC(C(=O)c2ccccc2)C(C)CC)c(OC)cc1Cl C(C(C)(O)CC(=O)NC1CN(C(c2cc(C(F)(F)F)nn2C(C)C)=O)C1)OC c1(C(N2CCC(O)(CCNC(CC(CC)C)=O)C2)=O)cn2ccc(OC)cc2n1 C(CCCC(C)C)(c1nnnn1Cc1ccccc1)NC(c1ccn(CC)n1)C C#CCC(CC(F)F)C(=O)N1CC(C)CN(C(=O)C(CO)CC(C)C)C(C)C1 C1(CCC)(NC(c2ccc(=O)n(CC)n2)=O)CCCN(C(=O)C(O)CC)C1 C12(CNC(C(CC)(C)C)=O)CC(NC(=O)CN(C)C(C)C)(C1)C(C)O2 C1(CC)C(C(=O)NC(CC(=O)N(C2CC(C)(C)C2)C)C2CC2)CCN1C N1(C(CC(C)OC)=O)CCCCC(NC(c2cc(F)ccc2Cl)=O)C1 C1(C(=O)NCC(CO)N(C)C)CCC2(CC2)N1C(c1ncc[nH]1)=O c1(C(N2CC(O)(CNC(C3(C)CC=CCC3)=O)C2)=O)ccc2c(c1)NCCC2 c1(NCCCC)ccc(C(=O)NC2(CNC(C3CCN(C)CC3)=O)CC2)c(Cl)c1 c1(C(=O)NC2C(n3cc(CC(C)O)nn3)CCC2)ccc2nncn2c1 C(=O)(CC(COC)COC)NC1(CF)CCN(C(C2CN3CCC2CC3)=O)C1 C1(OC)CC2CC(C(=O)NCCCNC(c3cn(-c4ccccc4Cl)nn3)=O)CC12 c1(C(N2CC3CN(C(=O)CCc4ccsc4)C3C2)=O)c(F)cc(F)c(O)c1F Cc1ccccc1SCC(=O)NC1CCCC1CNC(=O)CNC=O C1(CC(=O)NC(c2ccc(F)cc2)(C(=O)OCC)C)CCC(=O)NC1 C1(NC(COCCCC#C)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1(C)C Cc1cn(C(C)C(=O)NCCc2ocnc2CNC(C2CC2C)=O)cn1 N1(C(c2[nH]cc(C)n2)=O)CCN(C(c2ccc(CN(C)C)o2)=O)C2CC12 CC(C)(CCCNC(c1scnc1Cl)=O)C(=O)NC1CCC2CCC1C2 N1(C(c2ccsc2Cl)=O)CCN(C(C2C3CCCCCCC23)=O)CC(O)C1 N1(C(c2cc(OC(C)C)ncc2)=O)CC2CCCC2(NC(c2cncs2)=O)C1 C1(C)(C(=O)NCCC(C)N(C(c2cc(C)n(C(C)(C)C)n2)=O)C)CCC(=O)NC1 c1(C(N(C2CC(NC(=O)C(F)(F)C3CC3)C2)C)=O)cc(Br)c2[nH]nnc2c1 OC1(C2CC2)CCCN(c2cc(NCC(Cl)=CCl)nc(C(F)(F)F)n2)C1 c1(C(CNC(=O)CC#N)NC(COCCCCC)=O)cc(F)cc(Cl)c1 CCC(C)(CNC(C1(CNC(c2cnc(F)cc2C)=O)CC(=C)C1)=O)C(C)O CCCC(C)(CCC)C(=O)N1C2CCC1CN(C(C1C(C)C1C)=O)CC2 c1(C(=O)NCC23CCCN(C(COCCCC)=O)C2C3)c(C)ncn(C)c1=O c1(C(=O)NCC=C(C(=O)NC(CCOC)CO)C)cnnc(C)c1 c1(C(C2CC3CNCC3C2)=O)ncnc2ccccc12 N1(C(COCCCC)=O)CCCC2(C1)CN(C(c1cccnc1N)=O)C2 N1(C(=O)Cn2nccn2)CCC=CC1C(N1CCCCCC1)=O C1(CNC(C(C2CC(F)(F)C2)OC)=O)CCCCN1C(=O)CCCN(C)C(C)C N1(C(C(F)=CC)=O)CCC2(CC1)COC(CN(C(C(=O)NC)C(C)C)C1CC1)C2 Cc1cc(C)n2ncc(C(N3CCC(CO)C(NC(=O)CCC4CC4)C3)=O)c2n1 C1(NC(=O)C=CC2CCCCC2)CCN(Cc2nnc(O)nc2O)CC1F c1(C(=O)NCC(CNC(C2(C(CC)=O)CC2)=O)C)cn2cccnc2n1 c1(-n2c(-c3[nH]c4c(c3C)CCCC4)nc(C)n2)cc(Cl)cc2c1OCC2 c1(C(N2CCC(CC#C)C2)C(=O)NC(C)C)cncc(C(C)(F)F)c1 c1(OC)cc(N)c(C(=O)NC2(CCNC(c3cncnc3C)=O)CC2)cc1OC N1(C(c2cc(Cl)c(Cl)c(Cl)c2)C(=O)NC2(C)CC2)CC(C(F)(F)F)C(C2CC2)C1 N1(C(c2c(C)nc(C)s2)=O)CCC(CNC(=O)CSC(F)(F)F)C(C)C1 c1(OC)ccc(Br)cc1CSC1CCCC1.N12CCC(C1)CCC2=O C1(N(C(c2cnc(CC)s2)C(=O)NCCN2CCOCC2)CC)CCN(C)CC1 c1(OC)cc(C(N2CC(C(=O)Nc3c(Cl)cc(Cl)nc3Cl)C2)=O)cc2n[nH]cc12 C12CCCN1NC(=O)C(Cn1cccn1)NC2=O.c1(NC)cccc(C(C)=O)c1 Cc1noc2ncc(C(N3CCC(NC(C4CCC4)=O)CC3C3CC3)=O)cc12 Cc1cc(=NC(=O)Nc2ccc(-c3csc(=N)[nH]3)cc2)cc[nH]1 C=CCCC(C(=O)NCC(=O)OCC)NC(=O)C(C1CCC1)OCC Nc1ncc(Cl)cc1C(=O)NCCOC1CCN(C(C2(CF)CCOCC2)=O)C1 N#Cc1sc(=NCCC2CCN(C(c3cccc4c[nH]nc34)=O)C2)[nH]c1Cl Cc1cnc(C(N2CC3CC2C3C(=O)NCC2=NOC(C)C2)=O)c(F)c1 C1(CC)(NC(c2nnc(S)n2C)=O)CNC(=O)C1.N12CC(C)(C1)OCC2=O c1(C(=O)NCCN(C(c2c(C)cc(CO)o2)=O)C2CC2)c[nH]c2cc(Cl)ccc12 C(=O)(CCC(=O)c1cccc(F)c1)NCC1CC(C(F)F)(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2CN(Cc3cn[nH]c3)C2)cc(F)c(O)c(Br)c1 Cc1ccc2nc(SCC(=O)NC3CN(C(=O)CSc4ccccn4)C3)[nH]c2c1 c1(C(=O)NCC(C)(C)CC(=O)N(C(CF)CF)C)cccc2[nH]ccc12 C1(COC)(NC(=O)C(C)N(C)C)CCCN(C(c2ccc(SC)cc2)=O)C1 C1(NC(C(CCC)NC(=O)Cc2cccnc2F)=O)CCCCCC1CO N1(C(c2cc(C)oc2C)=O)CCN(C(C2CC3C(C2)C3(C)C)=O)CC1CC(F)F C1(C(=O)NC2(C)CCN(C(CCC(=O)N(C)C)=O)C2)C2CCC(F)(F)C12 C1(CNC(C2C(C)(C)C2)=O)CN(C(C2CCC(F)(F)CC2)=O)CC2(CCC2)O1 C1(NC(COc2c(C)cccc2)=O)CCN(C(=O)CCC2CCCO2)CC1C N1(C(C)=O)CS(=O)(=O)CC1C(N1CC2(CCN2C(c2cc3c(s2)CCC3)=O)C1)=O N1(C(CN2C(C)CCC2)=O)CCCCCC(NC(c2cnn3c2CCC3)=O)C1 C(=O)(CCCCC(F)F)N1C(CNC(C2N(S(C)(=O)=O)CCC2)=O)CCCC1 c1(C(=O)NCC(C)(C2CCC2)NC(CCSC)=O)ccc([N+](=O)[O-])c(C)c1 C1(C(N2CC(O)(C(C)NC(=O)COC(F)(F)F)C2)=O)CCc2ncsc2C1 CC(C)C(F)C(=O)NC1CCCCC1CNC(c1ncoc1C(C)(C)C)=O c1(C(=O)NC2C(CC=C)CCC2)c(CNC(c2ccc(CC)o2)=O)cnn1C CCC(CNC(=O)COC1CC=CC1)(CC)NC(c1coc(C(F)F)n1)=O C(=O)(C(CC(F)F)NC(c1c[nH]cc1C)=O)N(CC#C)CC1CCCO1 Cc1cc(C=CC(=O)NCC(CNC(C2C=CCS2)=O)CO)ccc1F C1(CC(=O)NCC(=O)NCC(=O)NC(C)Cn2ccnn2)OCCC1(C)C O=C(C1=NNCC(F)(F)C1)NC(c1ccc(Cl)cc1)c1ccc(F)cc1 N1(C(CNC(=O)OC)=O)CCCC12CCN(C(=O)C(c1ccc(Cl)s1)=O)C2 Cc1nn(C)c2sc(C(=O)NCC34CN(C(C5CC5C)=O)CC(F)(C3)C4)cc12.CC1CC1 N1(C(C=CCNC(C(C)N2CCC2)=O)=O)CC(CO)C(C)(C)C1 N1(C(CC(COC)C)=O)CCN(C(=O)C(=Cc2cccnc2)C)C(CF)C1 Cc1cc(SC2CCCC2(C)C)c(F)cc1[N+](=O)[O-] N1(C(C(C)(C)C2CCOCC2)=O)CC2(CCN(C(C3(C)CC3Br)=O)C2)C1 N1(C(c2c(OC)c(C)cs2)=O)CC(C)(C)CCC1CNC(C1C2CCCCC12)=O c1(C(=O)NC(COC)CNC(=O)CSS(C)(=O)=O)cc(C)sc1C C1(NC(N(CC)Cc2ccc(C)o2)=O)C2Cc3ccc(Br)cc3C12 n1(CC)nnnc1NC(COCC(=O)NC(C1CCOCC1)C)=O C1(O)(C(=O)NC(C)CC2CN(c3cc(O)nc(O)n3)C2)CCN(C)CC1 C1(C(=O)NCC2C(NC(C3CSCC(=O)N3)=O)CC2)CCc2nc[nH]c2C1 c1(NC(=O)NC(C)(CN2CCOCC2)C2CCOC2)ccc2c(c1)OCO2 C(=O)(CC(O)CN(C)CC1CC(F)(CO)C1)N(C1(C(=O)Nc2ccccc2)CC1)C N1(C2CN(C(C(N3CCC(C)C3)=O)=O)C2)CC(NC(=O)Cc2cnoc2)CC1=O c1(C(N(CCC(=O)NCc2ccn(C3CC3)n2)CCO)=O)cnnc(O)c1 c1(C(N2C(C(=O)NCC(=C)CC)CC2C)=O)cc[nH]c(=NC)c1 c1(C(=O)OC)cc2n(n1)CC(Nc1ccc(-c3cccnc3)cn1)CO2 C1(CNC(=O)C2=NOCC2)CN(C(C2CC(OC(F)(F)F)C2)=O)CCCO1 C1(C(N2CC(COC)(NC(=O)C(C)CC3CC3)C2)=O)CCCCC(F)(F)C1 C(C(C)(C)C(=O)NC1(CC(=O)NCCc2ncccc2F)CC1)OCC C1(NC(c2nc(C)n(C)n2)=O)CCC(C)(NC(=O)CC2CCCO2)CC1 N1(C(c2c(C)nc[nH]2)=O)CCC2(CC1)CC(C)N(C(=O)CN1CCC(C)C1)C2 C#CC1CN(C(C2CCC(C)(CC)O2)=O)CCN1C(=O)C(C)CCC(C)(C)C C#CCCC(O)C(=O)NCCCCNC(C1(Cc2cccc(Cl)c2F)CC1)=O C(=O)(C(C)CCC(C)(C)C)N1C(C(=O)NC(C(C)C)c2nc[nH]n2)CCCC1 c1(C(=O)NCC2(C)CCN(C(C3C(F)(F)C34CC4)=O)C2)cc2cnc(Cl)cc2s1 CN1CCCC1C=CC(=O)NC1CC(NC(C2CCCCC2n2cccc2)=O)C1 N1(C(c2cc(OCCCSC)ccn2)C(=O)NCC)CCOCCC1C(C)C C12(NC(Cn3ccc(C)n3)=O)CC1CN(C(c1cc(C3CCCC3)nn1C)=O)C2 N1(C(C(C2CCN(C(=O)CC3OCCC3(C)C)C2)C)=O)CCCC(CN(C)C)C1 O=C(C1=CC2CCCC12)NC1CCN(C(=O)C(O)Cc2cnc[nH]2)C12CC2 c1(C(N(CC(C)(C)CNC(=O)CC23CCCC2C3)C)=O)cc2ncccc2[nH]1 C(C)(C(C(C)C)NC(c1cnn(C2CC2)c1Cl)=O)NC(C=COCC)=O c1(C(=O)NCC(C)CN(C)C(c2cc(Cl)ncc2N)=O)cccc2nccn12 C1(C)(OC)CCC(C(N2CCN(C(=O)C(=O)N(C)C)CC2C)=O)CC1 N1(C(CC(C)(C)O)=O)C(CNC(=O)C(=Cc2cccnc2)F)CC2CCCC12 C1(n2cc(-c3c(C)ocn3)nn2)CCCN(C(C2CC3(C2)CN(C)C3)=O)CC1 c1(C(N(CC(C)C)CC(C)C)=O)cn(CCNC(=O)C(n2cccn2)C)nn1 C1(CNC(C(CC=CC)NC(c2nscc2C)=O)=O)COCC(=O)N1C C1(C(=O)NCC2(CO)CCCN(C(CC(C=C)C)=O)C2)CCn2c(C)nnc2C1 N1(C(COC2CCN(C)CC2)=O)CC2CN(C(=O)CN3CCOC3=O)CC12 c1(C(=O)NCC2(CNC(C3CC3C3CCCO3)=O)CC2)csc(Cl)c1 c1(OC)nc(C(=O)NCC(O)CN(C(=O)CC(=O)NC2CC2)C)co1 n1(N(C(=O)CSC(C)(C)C)C)cc(CCOCP(C)(C)=O)nn1 c1(C(C)C)ccc(C(NCC2CCN(CC(F)F)CC2)OC)cc1Cl CC1=C(C(=O)NCC(C)(C)C(=O)NCC(c2ccncc2)O)CCC1 c1(-n2c(C(C)(C)NCC(CC3CCCCC3)SC)nnn2)ccc(F)cc1 C(O)(C(=O)N=c1cc(C(F)(F)F)[nH][nH]1)c1nc(C)oc1.C12(O)CN(C1)CC2O N1(C(=O)OC(C)(C)C)CCC(OC(CC(F)C2CC2)=O)C1 N1(CCOC)CC(C(=O)NC2(COC)CN(C(C3CCC(=O)NC3)=O)C2)CC1=O N1(C(CC#C)=O)CC(NC(c2ccc(-n3cccn3)cc2Cl)=O)CC(C)C1 C1(C(=O)NC(c2ncc[nH]2)CC)C=CCN(C(=O)C(CO)N(C)C)C1 C#CCCC(=O)NC1(CNC(=O)CC(C)c2ccco2)CCOC1 c1(C(N(C)CC2N(C(C=CC(C)(C)SC)=O)CCC2)=O)cccc2c1CC(=O)N2 CC1CCC2(CO1)CN(C(=O)Cn1cc3ccccc3n1)C1COCC21 C1(CC(=O)N(CCCC)CCOC)CCN(C(C2CCOC2C)=O)C1(C)C c1(C(N2C(CNC(=O)CCCn3ccnn3)CC(F)C2)=O)cnc2n1CCC2 CCCCCC(C)CC(=O)N(C1CCCN(C(c2cnn(C)c2Cl)=O)C1)CCF c1(C(=O)NC(COC)C2CC2)ccc(-n2cc(C3CCCC3O)nn2)cc1 c1(C(=O)NC(C)CC2CN(C(c3cnn(C)c3C3CC3)=O)C2)ccc(F)cc1Cl C1(C(=O)NC2CCOC(CO)C2)(NC(=O)NCC2CC2)CC(F)(F)C1 c1(CN2CC3C(C(N4CC(F)(F)C(F)(F)C4)=O)(C3)C2)c(Cl)cc(F)cc1Cl C1(NC(=O)CN2C(=O)CCCC2=O)CN(C(c2ccoc2)=O)CC2CCCC12 [N-]=[N+]=NC1CN(C(=O)CC2CCN2C(=O)CSCC(F)F)CC1O n1(CCC(=O)NC2(CF)CCN(c3nnc(CC)o3)C2)c(=O)oc2ccccc12 Cn1cnc(CC(O)C(=O)NCCCCCNC(=O)C(C)(C)n2cc(Br)cn2)c1 CC(C)(C)CC(F)C(=O)N1CCOC(C(=O)NCCC(=O)NC(N)=O)CC1 N1(c2ccnc(OC)n2)CCC(C2CCCN(C(c3c(Cl)n[nH]c3C)=O)C2)C1 N1(c2ncc(C)cn2)CCCC(C2CCCN(C(=O)CN3CCC(C)CC3)C2)C1 N1(C(C2CC(C)(O)C2)=O)CCCCCCC1C(=O)Nc1cccc(O)c1 C1(F)(C(=O)NCC2CCC(=O)N2)CCCN(C(c2cccc(F)c2O)=O)C1 C1(C2CC2)(C(=O)NC2CC(CCNC(c3cnccn3)=O)C2)CCOCC1 C(=O)(CCC(O)C(C)(C)C)NC(C)Cc1nncn1C.C12CN(C1)C2=O Cc1cc(C)c(CC(N2CCC(CN(C)C(C3CCSC3)=O)CC2)=O)c(O)n1 N1(C(C2CC=CCO2)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc(O)cc1 c1(CNC(CC2C(C)CCN(C(=O)CCS(C)=O)C2)=O)cccc2ccnn12 C1(NC(c2cccc(Cl)c2)=O)CN(C(c2ccnc(S)c2)=O)CC1C(F)F Cc1cc(I)ccc1C(N1C(C(N2CCC(F)(CO)C2)=O)CC2CC12)=O c1(C(N(CCCCCC)Cc2ccccc2O)=O)cc(Cl)cnc1OC CCCCC(CC)C(=O)NCC(C(=O)Nc1ccc(C#N)cc1CC)C(C)(C)C c1(OC)ccc2c(c1)nc(CO)n2C.C12(F)CC(C1)NC2=O c1(NC2(CNC(=O)CC=C(Cl)Cl)COC2)cc2nn[nH]c2cc1[N+](=O)[O-] C1(C(N2CCN(C(CSCC(N)=O)=O)CC2CCO)=O)CCc2nnnn2C1 c1(CN2C(C(=O)Nc3ncco3)CCC2)c[nH]c2ncc(C(F)(F)F)cc12 C(=O)(CC1CS(=O)(=O)c2ccccc21)NCCNC(CC(C)OC)=O c1(C(=O)NC(C)CCNC(=O)CCNC(N)=O)cc2nc(Cl)ccc2o1 n1(CC=C)cc(C(=O)N(CC(C)CNC(C2CCN2C2CCCC2)=O)C)cn1 c1(C(N(C2CCCN(C(CCCNC(C)=O)=O)C2)C)=O)nccc2c[nH]nc12 c1(N2CCC(C)C(NC(c3ncc(C(F)(F)F)n3C)=O)C2)ccnc2ncnn12 N1(CCC2(C(=O)NC(c3ncc(C)s3)(C)C)CC2)CCCCCC(S(C)(=O)=O)C1 N1(C(C(C)C(C)O)=O)CCC(F)(c2cn(CC3CCOC3=O)nn2)CC1 CCCCC(C(=O)NCC1(F)CCOC1)NC(c1scnc1Cl)=O C1(NC(C2CC3C=CC2CC3)=O)C2CC(CN(C(=O)COC3CCC3)C2)C1CO N1(C(C(C)Oc2cccc(C#N)c2)=O)CCN(N(C)Cc2ccnn2C)CC1 C(CCc1cn(CCN2CCOCC2)nn1)(C(F)F)NC(=O)CN1CC2CC2C1 C(=O)(CC(C(C)(C)C)NC(C1CN(C)CCO1)=O)NCC(=C)CC C1(C(N2CC(OC)(CNC(c3conc3C)=O)C2)=O)CC2(CCC2)CO1 C1(CC)CCCCN(C(=O)COCCCOC)C1.C12(CC1)C(=O)N2 c1(N(C)C)ccc(-c2nc(CC3CCOCC3)n(-c3ccnc(Cl)c3)n2)nc1 c1(C(N2CCCN(C(c3cnc(C4CC4)s3)=O)CC2)=O)nccc2c1NCCC2 c1(C(=O)OC)ccccc1C(=O)NC(C)CCNC(c1ccc(CCF)cc1)=O c1(CNC(C=CCNC(C2CCC(C)S2)=O)=O)ccn2ncnc2c1 Cc1cc(O)ncc1C(=O)NC12CCN(C(c3cc(N)cnc3C)=O)CC1C2 N1(C(C(CSC)C)=O)CCN(C(=O)CC2CCC(C)C2)CC1CCO Cc1cc(Br)ccc1C1(C(=O)N(C)CCC2CC2)CC1 C1(CC(=O)N(CCN(CC)CC)C)CCCN(C(=O)CC2CC(C)(C)CO2)C1 N1(C(Cn2c(C)ccc2C)=O)CCCCC(NC(=O)CSCC(C)C)CC1 C(=O)(C(COC)CC(C)C)NCC(CCNC(C1(COC)CC1)=O)O N1(C(c2ccc(Cl)o2)C(=O)NCC(=C)C)CCC2(CCCN(C)C2)C1 CC1CCCC(CCNC(=O)CC2(N(C(=O)CCSC3CC3)C)CC2)O1 C123CCC(CC1)(C2)C(=O)NC1CN(C1)CC(=O)N3.Cc1sncc1.C1(O)CC1 C1(OC)CC12CCCCCC2.C(=O)(C(C)C(=O)NC1COC(=O)NC1)OC C1(CC(=O)NCC(CNC(CN2CCC(C)C2)=O)(C)C)SC2=NCCN2C1=O C(=O)(C(CC1CCOC1)NC(=O)OC(C)(C)C)N(CCCC)C(C)Cc1ccccc1 CC(CCC(=O)NCC1(O)CN(C(=O)CC2CC3CC3C2)C1)N(C)C c1(-n2cc(C3(C)CN(C(=O)CC4COC(=O)N4)C3)nn2)ccc(Br)cn1 CCCC(CCCO)C(=O)N1CC(NC(=O)C(C)=C2CC2)C(C)C1 c1(CC(N2CC(NC(C3(CCCC)CC3)=O)C2)=O)ccc2c(c1)CC2 N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CC(NC(c1cc[nH]n1)=O)CCO2 CC1(C(=O)NCC2CCCCN(C(c3cc[n+]([O-])cc3)=O)C2)CCCC(F)(F)C1 c1(NC(C2CCCC(NC(CCNC(C)=O)=O)C2)=O)cccc(F)c1Br Cc1c(F)ccc(C(N2CCCC3(NC(c4cnsc4)=O)CC3C2)=O)c1N CCC(C)(C)C(O)C(=O)N(CC(C)NC(c1ccc(C)c(OC)c1)=O)C CC1(C)CCC(CC(=O)NCc2cc(C(N3CCC(O)C3)=O)no2)O1 c1(NCCCC)nc(N(C)CC2(CCO)CC2)nc2ncn(C)c12 CC1(C)C(=O)NCCCN1Cc1cn(-c2ccc(F)cc2)nn1 C(=O)(C1CCCc2nc[nH]c21)NCC1(C)CCCN(C(=O)CCOCC(F)F)C1 c1(C(C(=O)NCCN(C(=O)CSC)C(C)C)N(CC)CC)ccccc1 CCC1=NOC(C(N2CCC(C)C2CNC(c2ccc(C)cc2)=O)=O)C1 C1(c2n(CCC(=O)OCC)nnn2)(NN2CCCCC2)CC2CCCC12.C1CN1 C1(C(=O)NC2(CC)CC(C)(C)C2)CC2CN(C(=O)C(C)CC(=O)OC)CC2C1 c1(NC(C)=O)ccc(C)c(C(=O)NC2CN(Cc3cnccc3Cl)CC2F)c1 CON1CCC(C(=O)NCCCCC(C)NC(=O)CC2=CCCC2)CC1 CC1CCN(C(C2CC(=O)C23CCC3)=O)CC1CC(=O)NC1CC2C=CC1C2 C1(C(=O)NCC(C)NC(c2ccc3nnc(O)n3c2)=O)CCc2nnc(O)n2C1 N1(C(c2ccn(CCOC)n2)=O)CCN(C(=O)C=C=C(C)C)CC1CCOC Cc1nc(C(=O)NCC2CC2CNC(c2cccn2C(C)C)=O)ccc1Br CC1=C(C(=O)NC23CC2CN(C(=O)C(c2ccccc2)C2CC2)C3)CCS1(=O)=O N1(C(C(C#C)(C)C)=O)CCC2(CCCN(C(=O)C(C)Sc3ncccn3)C2)CC1 C1(CCC)(NC(=O)C(C)COC)CCCN(C(=O)CCCc2n[nH]c(=N)s2)C1 c1(OC)cc(C(=O)NC2CN(C(=O)CN3CCC3C)CC2(F)F)cc(F)c1 CC(C)CC(C)C(=O)NCCCCC1CCN(C(=O)CCCC#N)CC1 c1(OC)cnccc1C(N1CCSCC1C(=O)NC(C)C(C)(C)O)=O CC1=CCC(C(N2C3CN(C(c4nc(Br)cs4)=O)CC23)=O)CC1 C1(CN(C)C(c2cc(C3CC3)ccn2)=O)COCCN1C(=O)C=CC=C(Cl)Cl Nc1ccc(F)c(C(N2CC(NC(=O)Cc3cnccc3Cl)C(O)C2)=O)c1 C1(C)CCc2ccccc2C1.S(=O)(=O)(C1(c2cn(CN)nn2)CC1)N(C)C N1(C(COCC(C)C)=O)CCC(NC(c2cc(Cl)cc(Cl)n2)=O)C(O)C1 C1(C(=O)NCC(=O)N(C)CC2(CCO)CC2)CCCN1C.CC(F)F n1(CC(=O)Nc2ccc(-c3n(C)nc(CO)c3)s2)nnc2c1CCCC2 CC1C(=O)NCCCN1C(=O)NCCN1CCN(c2ccccc2)CC1 c1(CC2(N(C(=O)C(O)CNC(=O)CC=CC(C)(C)C)C)CC2)ccncc1Cl c1(C(N2CCCC(c3cn(CCOCCOC)nn3)C2)=O)ncnc(C)c1C c1(C(=O)NCC(CNC(=O)CNC(=O)CC2CCO2)CO)nsc2ccccc12 N1(C(C(CC)C#N)=O)CC(CNC(c2sccc2Br)=O)CC12CCC2 NC(Cc1csc(Br)c1)C(=O)Nc1cncnc1 C1(N(C(C)=O)CC)CCCN(C(C)C(=O)NCC(c2ccc(Cl)cc2)C)C1 CC(CC(C)NC(c1cnc(S)[nH]1)=O)NC(=O)Cn1cnc(C(N)=O)n1 Cc1scnc1C(=O)NC1(C(=O)NCCN(C(N)=O)C(C)C)CCC1 C1(CNC(CCC(=C)C)=O)CN(C)CCN1C(c1cc(OC)cc(Br)n1)=O N#Cc1cnccc1CNC12CC(C(=O)Nc3c(Br)ccnc3Br)(C1)C2 N1(C(CC(CC)NC(C)=O)=O)CCOC(C2CN(C(=O)C(CCOC)OC)C2)C1 Cc1cc(Cl)cc(NC(C2CCC3CCC23)=O)c1CNC(=O)OC(C)(C)C C(N=C(NC1CCCCC1C)NC1CCC1)c1cc(C)oc1 c1(COC)ccccc1C(N1CCCC(CNC(c2cnnc(O)c2)=O)C1)=O C12(OC)CCCC(CC(NC(c3ccncc3Br)=O)C1)C2 c1(C(=O)NCC(c2cccc(F)c2)(C)C)ccccc1C1CC1(F)F c1(C(=O)OC)ccccc1C(=O)N(CC(O)CN(C(=O)CC1COC(=O)C1)C)C C1(NC(C2(Cc3ccc(C)nc3)CC2)=O)CC2(CCN(CCCF)C2)C1 c1(CC(N2CC(NC(C3CC(C)(O)C3)=O)CC(C)C2)=O)ccc(F)cc1[N+](=O)[O-] C1(C(N(C2CCCC2)CCC)=O)COCCN(CC2Cc3nccn3C2)C1 Cn1cc(C(=O)NCCCCC2CN(C3CCCS3)C2)c(C(C)(C)C)n1 C(=O)(CCC(C)(F)F)NCCCN(C(c1ncccc1CO)=O)CC CCC(C)(CNC(=O)C(C)(CSC)NC(=O)COC1CCC1)C(C)O N1(C(C#C)C)CCCN(C(=O)NCC2(CCOC)CCCC2)CC1 c1(C(=O)NCCCC(C)NC(c2cnc(C)o2)=O)cc(C)c2nc(C)cn2c1 C1(C(=O)NCC2(O)CN(C(CCc3nc(C)sc3)=O)C2)CCC(O)CC1 N1(C(CSC)=O)CCC2(COCC(CNC(c3cncc([N+](=O)[O-])c3)=O)O2)C1 c1(C(=O)OCc2c(C)cccc2)ccc2nc(S)[nH]c2c1 c1(OC)cnc(F)cc1C(N1CCN(C)CC1C(=O)NCC12CNC(=O)C(C1)C2)=O C(CNC(=O)C(C1CCCCC1)F)(CC(F)(F)F)NC(c1n(C(C)C)ncc1)=O CCC(C)CCCC(=O)NCC(C)CNC(c1cc2ccncc2[nH]1)=O C=CC1(CC(N2CCC(OCC)C2)=O)CN(C(c2csc(C)n2)=O)C1 Cc1ccc(C(=O)NC2CC(CNC(C3CC3C)=O)C(O)C2)c(C(C)C)n1 C(CC)(CC(=O)NC1CC1C1CCOCC1)N(C(c1ccc(CC)[nH]1)=O)C N1(C(Cn2c(C)ccn2)=O)CCSCC1C(=O)NCCC1CCN(C)CC1 c1(NCCNC(=O)OC)[nH]c(=NCc2scnc2C)nc2c1ncn2C(C)C C1(CNC(=O)C(O)Cc2ccccn2)CN(C(=O)C=CC=C(Cl)Cl)CC12CC2 N1(C(C(SC)SC)=O)CC2CC(C(N3CC4(CCN4C)C3)=O)C(C2)C1 C1(CNC(c2c(CNC(=O)CC3CC=CCC3)cco2)=O)CC1C1CCC1 N1(C(c2nnn(C)n2)=O)CCC(NC(=O)COCc2ccccc2F)CC1 c1(CN(C(C2CC(O)CN2N)=O)CC)cc(F)ccc1F Cc1c(Br)ccc2c1CCC2NCc1ccc(F)c(C(F)(F)F)c1F N1(C(CC=C)=O)CC(C2CCCCN(C(C3CCOC3C(F)(F)F)=O)C2)C1 N1(C(C(C)n2ccnc2)=O)CCN(C(=O)CO)C2CCCCC2C1 c1(C(=O)NC2CN(C(Cc3ccc(C)nc3)=O)CC2C)cnc2c[nH]nc2c1 c1(CC)ncnc(CC)c1C(=O)NCCC1(NC(=O)CC2COC(C)(C)C2)CC1 C1(C(F)F)(OC)CCCN(C(=O)CCc2ccc(Br)c(F)c2)C1 C(CN=c1ccc(S(=O)(=O)N2CCN3C(=O)CCC3C2)c[nH]1)N1CCC(OC)C1 c1(OCC)ccccc1N(C(=O)C(=O)C(C)C)C(=O)CN1C(CO)CC2CC12 C1(NC(C(Cc2ccsc2)NC=O)=O)CC2(CCN(C(C3(F)CC3)=O)CC2)C1 C#CC(C)(C)C(=O)N1CC(CCNC(=O)CNS(=O)(=O)C2CC2)C(C)C1 c1(NC(C2(c3ccc(-c4cccc(SC)c4)cc3)CC2)=O)nc(F)ccc1Br NS(=O)(=O)c1ccc(CNC(=O)C(=O)NC2CCCN3CCCCC23)cc1 c1(C(N2C3C(c4cn(CCOCC)nn4)C(C3)C2)=O)c(O)ccc(OC=O)c1F Cc1nc2c(C(=O)NC3C4CC3N(C(c3cc(C)sn3)=O)C4)ccnc2[nH]1 Cc1ccc(SCC(N2CCCCC2CCCNC(=O)CC2CC23CC3)=O)cc1 Cc1ccc(F)c(C(=O)NCC2CC2NC(c2cnnc3ccccc23)=O)c1Cl c1(CCC(=O)NCC(CC)NC(=O)C(C)C(F)F)c(C)noc1C Cc1ccc(OCCN(C)CC2CCN(C(c3nc(C)n(C)n3)=O)C2)cc1 CCCCCC(C)(C)C(=O)NC1CC2CC(C1)N(C(=O)CCOCC(C)C)C2 C12(C(N3CCCC(CCOC)C3)=O)CCCC1CCN2C(C1SCC=C1C)=O CC(CNC(C1(C)C=CCCC1)=O)CC(=O)N(C1CCCC1(C)O)C Cc1coc(C)c1C=CC(N1CC2CC(NC(C3CC4C=CC3CC4)=O)C1C2)=O N1(C(C(C2CCOCC2)C)=O)CCC(NC(C2CC(N(C)C)C2)=O)C12CCC2 c1(C(=O)NC2(C(C)C)CCC2)cccnc1CNC(=O)C(F)CC1CCOC1 Cc1nc2ncc(C(N3CCCC3CNC(=O)CCCCC#N)=O)c(=O)n2[nH]1 N1(C(c2ccc(OC)cc2Br)=O)CCCC2C1CCN2C(c1ccnc(O)c1)=O C(CCCCC(=O)N1CCCC(F)(NC(C2(CO)CC2)=O)C1)OC.c1ccccc1 Cn1c(C(=O)NCC(=O)NCC(N2CC(C#N)C2)=O)cccc1=O C(CCCCC(=O)N1CCC(O)C1(C)C)NC(CC=CC(C)(C)C)=O C=C(Cl)CC(C(=O)NCC(C)C1CCC1)NC(=O)C(F)OC(F)(F)F Cc1c(NC(C)C)cccc1C(N1CCOC(CNC(c2cncs2)=O)C1)=O c1(CN=c2cc(C3(O)COC3)nc[nH]2)cc(O)n2nccc2n1 c1(CSCC)ccc(C(=O)NC(C)(C)C(C)NC(=O)Cc2nonc2C)cn1 N1(C(CCCOCCOC)=O)CCC(N=c2[nH]c3ncc(Cl)cc3s2)C(C)C1 C1(C(=O)OCC)CN(C(C2CC3C=CC2O3)C(=O)NCCOC(C)=O)CCO1 N1(C(C(C=C)c2ccccc2)=O)CCC2(CC1)CN(C(c1cc(S(N)(=O)=O)co1)=O)C2 c1(C(=O)NC2C(C)CN(C(c3cccnc3C3CC3)=O)C2)cnn2ccncc12 CS(=O)(=O)c1ccc(CCC(C2CCC(F)(F)CC2)CO)cc1 N1(C(c2cc(C)c(Br)s2)=O)CCC(F)(CNC(C2CCOC2)=O)CC1 C1(C(=O)NC23CC(NC(C4(C(F)F)CC4)=O)(C2)C3)C(C)C1(C)C.CCOC Cc1ccc(CN(C)C(C2C3CN(C(c4cnc(Cl)s4)=O)CC23)=O)nc1 Cc1csn2ncc(C(=O)N(CC(CO)(CO)NC(c3ccoc3)=O)C)c12 N1(C(C2CCC3CCCCN23)=O)CCCC2(CCN(C(=O)CC3CC3)CC2)C1 N1(C(=O)Nc2ccc(N(C(C)=O)C)cc2)CCC2OC(=O)OC2C1 C(CCCCC(=O)N1CCN(C(=O)C(O)C(F)(F)F)C(C2CCC2)C1)=CC N1(C(CC2N(C(C=CCCCC)=O)CC2)=O)CCn2nc(C)cc2C1 N1(C(C2CCC(CC)O2)=O)CCC(C)(C)C(C(=O)NC2CC(C)(O)C2)C1 N#Cc1ccnc(N2CCCC(C(=O)NCc3cccs3)C2)c1 N1(C(C(CSC)O)=O)CCc2nc(CNC(C3CC4CCC(C3)S4)=O)sc2C1 c1(CNC(C(=O)Nc2ccc(OC)c(Cl)c2)=O)ccc2sc(=O)n(C)c2c1 C(=O)(CCCCN=[N+]=[N-])NCc1occ(C(=O)NCC2N(C)CCN(C)C2)n1 c1(C(N2CC(C)N(C(=O)Cc3ccsc3)CC2C)=O)ccc2ccccc2c1 C1(NC(C(C)(F)F)=O)CN(C(=O)Cc2cccc3nsnc23)CC2(CC2)C1 c1(OC)cc(OC)c(OC)cc1N(C(c1ncn(C)c1Cl)C(=O)NCC1CC1)C c1(OCCOC)cc(C)cc(CNC(=O)Cn2cccc2)c1C S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NC(c1cc(Cl)cc(Br)c1)CC(=O)O O(C1CCc2c(Cl)ccnc21)C(C1(Cl)C(C(=O)O)C1)=O C12(NC(c3cnc(CNC(C45CSCC4C5)=O)nc3)=O)CCN(CC1)CC2 C(CCCCCC1CC1)NC(=O)CCCn1cc(C2CC=CCC2)nn1 C(=O)(C(C)(C(F)F)c1ccccc1)NC1N(C(CCc2c(C)n[nH]c2C)=O)CC1 N1(C(c2ncc(N)nc2)=O)CC(NC(=O)CC2(O)CCC2)CC12CCC2 Cc1cc(=NCCP(C)(C)=O)[nH]c(N2CC3CC(C)(C)C3C2)n1 c1(CC)ccc(F)cc1C(=O)NC1C=CCN(C(=O)C2=CCCCC2)C1 CCCC(O)C(=O)N1CCOCC1CC(=O)NCc1ccoc1C(N)=O c1(C(N2CC(C)C(NC(c3ccc(Cl)nc3O)=O)C2)=O)cnc2c(c1)CCCO2 Cc1ccc2c(c1)CCC(C(N1CCC(C)(CCNC(C3CSC3)=O)C1)=O)O2 N#Cc1ccc(-c2cn(CC3CCN(C(=O)CCCCCF)C3)nn2)cn1 Cc1ccc(C(=O)NCC(CO)NC(=O)Cc2ccccc2CC(N)=O)c(O)n1 N1(CC)CC(NC(c2c[nH]nc2CNC(C2(C)CC3(CCC3)C2)=O)=O)CCC1=O CC1COCCC1NC(=O)OC(C)(C)C.c12ccccc1CC(=O)N2 C(CC(C(=O)N(C)CCOC(CC)CC)NC(c1cccc(O)n1)=O)OC Cc1cccc2c1CN(C(=O)CC(CNC(=O)C=Cc1ccc[nH]1)C1CCC1)C2 C1(NC(C(c2cccs2)NC(CCNC(COC)=O)=O)=O)CCOC2(CCC2)C1 c1cc(CC2CC2)c(C)o1.N1(CC)CC(C(=O)NC2CC(C(=O)OC=O)C2)CC1=O c1(C(N(C2CN(C(=O)CC3CCC3)CC23CC3)C)=O)nc2c(s1)CN(C)CC2 N1(C(c2ccc(CN(C)C)o2)=O)CC2(C1)CN(C(C1CCCO1)=O)C2 c1(OCC2CCCN(CCCCS(=O)(=O)N(C)C)C2)cc(F)cc2c1OCOC2 C1(C(=O)NCCCN(C)C2CC2)COC2(C1)CN(C(c1nc(Cl)cs1)=O)C2 CC12CN(C1)C2.c1(CNC(=O)CC2CCC2)ccn(CCF)n1 C1(CNC(C(C)(C)OCC)=O)CC2(CC(NC(=O)CN3CC4CC4C3)C2)C1 Cc1cccc2nc(C(=O)N(CCC(C)NC(c3cc([N+](=O)[O-])c[nH]3)=O)C)cn12 c1(C(=O)NC23CC(NC(=O)CC4COCCO4)(C2)C3)cn2ncccc2n1 c1(C(=O)NC2CC3C(NC(Cn4ncc(CC)c4)=O)C3C2)cc(C)c(O)nn1 c1(OC)cc(N)c(F)cc1C(=O)NC(C)CNC(c1cccc(C2CC2)c1C)=O Cc1c(C(=O)NC(C)CCCCNC(=O)CN(C)C2CC2)nnn1C1CCOC1 C1(C(=O)NCC(C)NC(C2(SC)CCC2)=O)Cc2nnsc2S1 C(C)(C)(CC(=O)NC1CC(N2CCCC2)C1)N(C(C(=O)NC)=O)C Cc1cncc(C(=O)NC2CCC(N(C)C(c3cc(Br)co3)=O)CC2)n1 N1(C(c2c(OC)n(C)nc2)=O)CCC2CC(C1)CN(C(=O)CC1CCCC1)C2 c1(C(N2CCCC(NC(=O)Cc3cnccc3Cl)C2)=O)cnc2scnc2c1 C1(C(=O)NC(CN(C(c2c(NC)cccn2)=O)C)C)CC2CCCCCC12 CC1(C(N2CCCC2CNC(c2c(Cl)ccc(F)c2F)=O)=O)CCC(F)(F)CC1 N1(C(c2c(C)sc(C)c2Br)=O)CCCC12CCN(Cc1ccccc1)CC2 C(CN=c1[nH]cnc(C)c1F)OCCN(C(CC(CCCCC)C)=O)C C1(C(=O)NC2CC2C(=O)NCCOC(F)(F)F)CCCCCCC1 N1(C(C(CC)CC)=O)CC2CS(=O)(=O)CC2(NC(=O)C(C)OC)C1 C=CCC(Cc1ccccc1)C(=O)N1CCCCC1CCNC(=O)C(=O)NCC Cc1nccc(CCN(C2CCCC2)C(C2CC3CNC2C3)=O)n1 N(C(=NCCF)NCC(c1cc(C)on1)(C)C)C1N(CC)C(=O)CC1 C(=O)(C(C)CC(F)(F)F)N1CCC(N(C23CCC(CC2)C3)C(c2c(C#C)c[nH]n2)=O)C1 O=C1NC(C2CC(=C3CCOC3)C2)C(=O)N1CC1CCC1 C1(CCNC(CCC=C)=O)CN(C(=O)Cc2ccc(OC)cc2)CC(C)O1 N1(C(c2ccc(C)c(O)c2)=O)CCC(C2CCN(C(=O)C(C)C(C)C)CC2)CC1 C1(NC(C2(n3ccc(C)n3)CC2)=O)CC2CN(c3nc(C4CCCC4)ns3)CC2C1 C123CCC(CC1)(C2)NC3=O.N1(N2CC3C(CO)C3C2)CC2CCCC2C1 C(=O)(C(C)(F)CC1CCCC1)N1C(C(C)NC(c2scnc2C(F)F)=O)CCC1 c1(C(N2CCC(NC(C3(CC)CC3)=O)CC2C)=O)cc2ccc(Br)cn2n1 N1(C(c2nccc(OC)c2)=O)CC(F)(F)CC1(C)CNC(C1CCC(F)(F)C1)=O C1(NC(c2cc(-c3cnn(C4CCOCC4)c3)[nH]n2)=O)CCS(=O)(=O)NC1 C1(N(C(=O)C(C2CCCCC2)NC(=O)CCCn2cncn2)C)CCOC(C)(C)C1 Cc1ccc2c(O)c(C(=O)NCC3CC4CC(=O)C3C4)cnc2n1 C1(NC(CNC(CCC)=O)=O)C(C)CCN(C(c2cnn3cccnc23)=O)C1C C12(C(N3C(C(C)O)CCC3)=O)CCC(CN(C(=O)C=CC3CCCCCC3)C1)C2 Cc1ccc(C(N2CCCCC2CNC(c2nc(Br)c(C)s2)=O)=O)c(O)c1 N1(C(CSCC#C)=O)CCOC2(CCN(C(=O)CC3(OC)CC3)CC2)C1 C1(NC(C2N(CC(C)C)CCC2)=O)CC2(C1)CC2NC(=O)Cc1cc[nH]n1 C1(C(=O)OC)CC2CC1CC2NC(C(=O)O)C1(C)CC1 c1(C(N2CCC(NC(=O)CN3CCS(=O)CC3)(CO)C2)=O)ccc2n[nH]cc2c1 C#Cc1ccc(C(=O)N(C2CCCN(C(c3cc(C)c[nH]3)=O)C2)C)cc1 Cc1noc(C)c1CCC(=O)NC(CO)C(C)NC(=O)CC(O)CN(C)C N1(C(C2CCCC(C(N)=O)C2)=O)C2CCC1CN(C(C1CC3(CC3)CO1)=O)C2 C1(NC(C(c2cccs2)SC)=O)CC2CCCC(C1)N2C(=O)C=CC1CCCO1 C1(O)(C(C)NC(C2(c3ccncc3)CC2)=O)CCN(C(=O)C(C)(F)F)C1 c1(OC)ccc(Cl)c(C(=O)NCC(c2cccc(C)c2)NC(=O)C2=CCC2)n1 CCC(C)CC(=O)C(=O)N1CCC(NC(=O)CN(C(=O)OC)C2CC2)C1 C1(CNC(c2ccc(O)nc2)=O)CCCN(C(c2cnn(CC(F)F)c2)=O)C1 CC1CCN(c2nnc(-c3ccccc3)o2)CC12CCC2 N1(C(C)=O)CCCCC1C(=O)NCCC(O)CNC(c1n[nH]cc1C1CCC1)=O C12(NC(c3nc(C4CN(C(c5nc(O)n[nH]5)=O)C4)oc3)=O)CC=CCN1CCC2 Cc1cc(C)cc(C=CC(=O)NC2CCN(C(=O)C(F)(F)CO)C2)c1 CC1CCC(NC(=O)C2=CSCS2)CN1C(=O)COC1CCOCC1 N1(C(c2ccc(C)cc2)=O)CCCC(C)(CNC(C2CNC(=O)O2)=O)C1 C(=O)(C(C(C)C)C1CCC1)N1C(CCC2CCCN2)(OC)CCC1.C(C)=O c1(C(c2nnnn2C(C)C)NCCC(CCSC)O)cc(Br)ccc1I C1(C(=O)NC2C3(NC(C=COCC)=O)CCC(C2)C3)CC2(CCCCC2)S1(=O)=O n1(CC(=O)NC(C2CC2Br)C)ccc(C2CC2)n1 CCCC(CC)CC(=O)N(C1CC2CCC(C1)N2C(C1CCC(C)(C)CO1)=O)C c1(CC(N2CCC(C(C)NC(C=C(CC)C)=O)C2)=O)ccc(OC(F)F)cc1 C1(C)(CC)CCC(C(=O)NCc2cc(C(N3CC(c4nncs4)C3)=O)co2)O1 c1(C(=O)NCC2C(C)(C)N(C(=O)CCC3CCC3)CC2)cccc2oncc12 c1(C(N2CCC3(CC2)CC3NC(C2(O)CC2)=O)=O)c(O)cnc2cc(F)ccc12 c1(OC)cc(C(=O)NC(C)C(C)NC(c2cc(Cl)c(F)cc2N)=O)cc(F)c1F c1(C(=O)NC2C(C)CCN(C(CCCC)=O)C2)ccc2c(c1)CN(C)C(=O)N2 CC1OC2(C(N3CCC(C(C)NC(c4cc(=O)cc[nH]4)=O)C3)=O)CCC1CC2 C1(CCC=C)CCCN(C(=O)C(CN(C)C)NC(=O)CC(CC)OC)C1 N1(C(C2CCC(O)C2)=O)CCC(CNC(=O)CC2(CO)CCCC2)C(F)(F)C1 c1(C(=O)NCC2CN(C(c3cc4c[nH]nc4s3)=O)CC2O)cccc2sccc12 C12(C(N3CC(C(=O)NCC4CN(C(C)=O)C4)OCC3)=O)CCC(C)(C1)OC2 C1(CC(=O)NC(CC)C(C)O)Cc2ccccc2CN1Cc1ncc(Br)cc1Br Cc1cc(C(=O)NC(Cc2ccoc2)C(=O)N(CC(=O)N(C2CC2)C2CC2)C)cs1 c1(C(N(C2CCN(C(=O)COC3CCSC3)C2)C)=O)cnn(C2CCOCC2)c1 N1(C(c2cc(C)c(F)cc2)=O)CCC(F)(F)C(C(=O)NC2CCCN(C)C2)C1 C(=O)(C1=CC2CC=CCC12)NC1COCCN(C(Cc2c(C)nn(C)c2)=O)C1 S(=O)(=O)(c1ccc(C(=O)NC(C)(C)CCNC(=O)CSc2nncs2)cn1)NC c1(C(=O)NC2C(NC(Cc3nc(COC)sc3)=O)CC2)ccn2nnnc2c1 CN1c2ccccc2CC1C(=O)NCC12CC(CN1C(C1CC(N(C)C)C1)=O)C2 c1(C(N(C2CCN(C(C3CCCC(=O)N3C)=O)C2)CC)=O)ccc(F)c(C)c1 c1(C(N2C(CNC(c3cc(OCC)no3)=O)CCC2)=O)ccc2c(c1)NCC2 Cc1ccnn1CC(=O)NC(Cn1ccnn1)C(=O)NCCCNC(N)=O C(c1ccccc1C)=CC(=O)NC1CN(C(CCC#C)=O)C1 N1(C(C(C(C)C)N(C)C)=O)C2CCCC1CN(C(c1csc3cncn13)=O)C2 C(=O)(C1=CC(O)CCC1)N1C(CCCNC(C=C(C)c2cccs2)=O)CCCC1 CC(C)(F)CCC(=O)NCCc1cn(-c2ccc(F)cc2C(F)(F)F)nn1 N1(C(C2(C)CCN(C(C)=O)C2)=O)CCC2(CCC(NC(=O)C(C)C3CCC3)C2)C1 CCCC(C)N=c1[nH]c2c(c(=NCCCc3ccc(Br)cc3)[nH]1)CCCC2 C1(C(N(C2C(NC(C(C)NC(N)=O)=O)CCCC2)CCO)=O)CCC2(CCC2)C1 N1(C(CC(C(C)C)O)=O)CC2CCC1CN2C(c1cc(C(F)(F)F)cc(O)n1)=O N1(C(C(C)(C)NC(C)=O)=O)CCCCC1CNC(=O)C(c1ccc(F)cc1)C c1(C(=O)NCC2(NC(c3nc(OC)oc3)=O)CCCC2)cc(F)cc(Cl)c1O C1(CNC(c2cc(CCC)nn2C)=O)CN(C(=O)C#CC(C)(C)C)CCCO1 c1(N(C)C)ccc(CN2CCCC(CNC(=O)C(c3ccccc3)O)C2)cc1 c1(CC(=O)NCCC(C)NC(C(COCC)C)=O)cccc(C)c1Br C1(N(C)C)C=CCN(CC(=O)NCCCN2C(=O)CCC2=O)C1 n1(CC)nc(C(N2CCC(C3CCCN3C(=O)Cc3csnn3)C2)=O)cc1O N1(CC(N2C(C)(CNC(c3csc(Cl)c3Cl)=O)CCC2)=O)CCS(=O)(=O)CC1 c12ccc(cc1)S(=O)(=O)N2.C12(CNC(CCC)=O)CC1CN(C(C1CCCC1)=O)C2 C1(NC(C2CCN(C(C(C)(CO)CO)=O)CC2)=O)CS(=O)(=O)C12CCC2 CCC(O)C(C)C(=O)N1CCC(C)(CNC(=O)C(C)Cc2ccc(F)c(F)c2)C1 C1(CNC(c2cc(Cl)c(F)c(Cl)c2)=O)CN(C(c2cccnc2)=O)C2(CCC2)C1 C12(CNC(c3c(SC)cccc3)=O)CCC1CCN2C(c1[nH]cc(C)c1C)=O Cc1ccc(CNC(=O)C(CCSc2cc(CC(C)C)on2)NC(N)=O)cc1C C12(C(=O)NC3CN(C(c4nc(C)oc4C)=O)CC3C)CC(CC(C)O1)C2 c1(C(=O)NCC(C)N(C(C(COC)OC)=O)C)cnc(-n2cccn2)c(C)c1 C(=O)(C(C)(F)C(=O)NCc1cc(C)c(C(=O)NCC2CCCCS2)o1)OC c1(C(N2CC(CCn3cc(C(CC)(C)C)nn3)C2)=O)nnn2c1COCC2 C(=O)(CCCCC(=O)N(C)C)NCCC(C)N(C(c1c(SCC)cccc1)=O)C N1(C(C2(CCOC)CCC2)=O)CCC(O)C(NC(=O)C(C)OCC(C)C)C1 C1(C2CC2)(C(=O)NC(CC#C)C(=O)N2CCCC(CO)C2)CC(=O)C1 C1(NC(C2C(OC)CCC2)=O)CCC2CCN(C(c3nc(O)c(C)s3)=O)C1C2 N1(C(C(CC)OC)=O)CCCN(C(c2cccc3c2OCO3)=O)C(C)C1 C(c1cnccn1)=CC(=O)NCC(C)NC(C1CC(=O)C1(C)C)=O Cc1cc(C(=O)NC2CC(N(C)C(c3cc(C(C)C)on3)=O)C2)c2occc2c1 c1(NC)ccc(C(N2CC(NC(=O)C=C(C)c3ccsc3)C3CC23)=O)nc1 CCCC(C)CC(=O)NC1COCCC1NC(c1cccc(OC)c1C)=O c1(C(N2CC(COC)(NC(c3ccc(OC)cn3)=O)C2)=O)cccc(C)c1O Cc1ccc(C(=O)Nc2cc(CC3CCCCC3C)cc(F)c2)c2ncccc12 N1(C(c2cc(C(=O)OC)[nH]n2)=O)CC2CC(C1)N(C(C1CCC3(CC1)CC3)=O)C2 C(=O)(C1=CCCCO1)N1CC(C(C(=O)NC(C=C)C(F)(F)F)OC)C1 c1(C(C)C)ncc(Cl)c(C(=O)NC2(C)CCN(C(c3nocc3C3CC3)=O)C2)n1 N1(C(C=COCC)=O)CCCC2(C1)CN(C(c1cc(C)ccc1C)=O)CCO2 C1(NC(CC)CCc2ccccc2)CN(C)CCN(C)C1 C(C)(C)(C(C)CC(=O)NC1(C)CCCCC1)NC(COC)=O Cc1c(C(=O)NCC2CN(C(=O)C3CC3)CC23CCC3)oc2ccccc12 C1(NC(C(n2ncc(C)c2)C)=O)CCOCC1NC(=O)C=CC(=O)NC1CC1 C12(C(=O)NCCCCN(C(c3ccc(CCC)s3)=O)C)CC1COC2(C)C C1(C(=O)NC(CC)(CNC(=O)CC2CCCC2)CC)COc2ccccc2C1 N1(C(C(C)NC(N)=O)=O)CC2CCC1CN2C(C12CCCC1(C(N)=O)C2)=O C=CCN=C(NCCOC(COCC(F)(F)F)=O)N1CCC2C(C1)NC(=O)N2C C(CCC(=O)NCCCCN1CCCC1)NC(C(C)OCC#C)=O C1(C(C)C)CCC(C(=O)N(C)CCN2CCCC2)C(=O)N1 Cn1cc(C(=O)NC2C3CC2N(C(=O)CC2CC(O)C2(C)C)C3)cc1Br c1(CC(=O)NCCSCC(=O)NC2CC(C(F)(F)F)C2)cccnc1 N1(C(c2cc(Cl)c(F)cn2)C(=O)NCCCC)CCC(P(C)(C)=O)C1 C(=O)(CCS(=O)(=O)CC(C)C)NCC1(C)CCN(C(C(C)OCCCC)=O)C1 C(C(=O)Nn1nnc(C)c1C)N(CCC(C)C)C(C1CC(CC)(CC)C1)=O N1(C(C2CCN(C)CC2)=O)CC(N=[N+]=[N-])CC1C(N1CC(O)C(C)(C)C1)=O c1(OC)ccc(C(N2CCN(Cc3ccc(OC)nn3)C(C(C)C)C2)=O)c(Br)n1 c1(C(N2CC3C(=O)NC(=O)C3C2)C(=O)NCC(F)F)cnc2ccc(F)cn12 C(=O)(C(C(C)(C)C)NC(N)=O)NCCC(C)NC(CSc1ccc(OC)cc1)=O Cn1cnc2[nH]c(C(=O)NC3(CNC(C4CCC(C#N)C4)=O)CCCC3)cc12 CCCCCC(CC)C(=O)NCC12CC(NC(c3cn(C(C)C)nc3C)=O)(C1)C2 C(CCCCCCO)NCCNC(c1ccccc1F)CC(=O)OC Cc1c(NC(=O)C(=O)Oc2ccnn2C)cccc1CSC(C)C C(=O)(C(C)(C)CO)NCc1c(C(N(C)CC2CC2(F)F)=O)occ1 c1(NC(=O)NC2(CSc3ccnc(F)c3)COC2)cccc(I)c1 c1(CC(=O)NC(C2CC=CCC2)C(=O)NC2(CC)CC2)cnc(O)cc1C CC1CCC(C(=O)NCC23CC2CN(C(C2CCN(CC4CC4)CC2)=O)C3)CC1 N1(C(c2nnc(C)o2)C)CCc2ccccc2C1CNC(C1(F)CCOC1)=O c1(OC)cc(N)c(F)cc1C(N1CC(NC(c2cc(C)co2)=O)C2CC12)=O c1(N2CCN(Cc3c(C)cc(C)[nH]3)C3(C2)CC3)ncnc2ccc(F)cc12 c1(OC)c(Cl)cc(C(=O)NCCN(C(c2nc(Cl)cs2)=O)C2CC2)cc1Cl CCC1=C(C(=O)NC2(C3CCN(C(=O)C(C(C)(C)C)OC)CC3)CC2)CCCO1 C1(S(N)(=O)=O)(C(N2CC(C)C(CNC(=O)C3=NNC(C(F)(F)F)C3)C2)=O)CCC1 c1(C(N2CC(C)CC(NC(C3=C(C)CCC3)=O)C2)=O)cn2nc(C)sc2n1 N1(C(C(C=C)O)=O)CC2CC(NC(=O)Cc3cccc(COC)c3)CC2C1 Cc1csc(CCCC(=O)N2CCC(C(C)NC(=O)CSC(F)F)C2)n1 N1(C(C(N2CCC(C)CC2)=O)=O)CCC=C(CNC(C2CC(O)C2)=O)C1 c1(C(N2CC(OC)(CNC(=O)Cc3ccnn3C)C2)=O)ccc(C(C)F)cc1 N1(C(Cc2nc(C)oc2)=O)C(C)CN(C(C23CC(C)(CCO2)C3)=O)CC1C c1(CC(=O)OCC)cccc(NC(C2CN(C(C3(Br)CC3)=O)CCO2)=O)c1 c1(OC)cccc2c1CCC2NC(=O)CCN1CCCS1(=O)=O N1(C(CN(CCOC)C)=O)CC(NC(=O)C=Cc2ccc(OC)cn2)C(C)(C)C1 C(=O)(CC1OCc2cc(Cl)ccc21)N(CCN(C(C1(CC=C)CCOC1)=O)C)C n1(CCCC)nnnc1C(c1[nH]cnc1C)NCc1nncn1CC c1(C(N2CCCC(CC(N3C(C)(CCO)CCC3)=O)C2)=O)ccc2c(c1)OCC2 C(C(C)(C)CO)(C1CC1)N.c1(CC)cc(C(N2CCC2C(=O)NCC2CC2)=O)n[nH]1 N1(C(c2cnc(C)s2)=O)CC2CC1CN(C(c1cn(C)cc1C)=O)C2 c1(NCCc2ccc(C)cc2C)[nH]c(=NC2CC3C(C2)C3(F)F)nc2scnc12 c1(C(N2CCN(C(C(CCC)NC(N)=O)=O)CC2C)=O)nc2ncc(C)cn2n1 C(=O)(CCC(=O)NC(C)CCN(C)C(c1sccc1OC)=O)NC N1(C(CN(c2ccccc2)CC)=O)C2CCC1C(CNC(c1cnc(C)[nH]1)=O)C2 Cc1nn(CC(=O)NCC2CN(C(=O)CCCn3cncn3)CC2C)c(=O)o1 c1(C(=O)NCC(C)(C2CC2)NC(c2c(CCC)[nH]cc2)=O)c(C2CC2)noc1C c1(C(=O)NC(CNC(C(C2CC2)SC)=O)CO)cccc[n+]1[O-] c1(C(=O)NCC2(F)CC(NC(c3ccc(N)cc3O)=O)C2)ccn2ncccc12 c1(C(=O)NC(CNC(C2CC3CC3C2)=O)C2CC2)c(F)ccc2nc[nH]c12 c1(OC)ccc(C2CC2C(C)NCCc2cc(C)n(C)n2)cc1 C1(NC(C2CC23CCC3=O)=O)CC12CCCCCC2 Cc1cc2cccnc2nc1C(=O)NCCNC(=O)CN1CCC(N(C)C)CC1 CCC(C)C(=O)NCC(=O)NCC1(C)CC(NC(C2CC(C(F)(F)F)C2)=O)C1 C1(NC(C2C(C)C2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)C2(CCCCC2)C1 C1(NC(C2C(C)C2)=O)CCN(C(c2ccc(-n3nnnc3O)cc2)=O)CC1(C)C Cc1c(C(C)NC2(c3nnnn3C3CCCCC3)CC(C#N)C2)cnn1C C1(C(N(CC(=C)C)C)=O)CCCCCCN1C(C1C2(CC2)C12CC2)=O C12(NC(c3cccc(C)c3)=O)CCC(C(=O)Nc3nc(S(C)(=O)=O)cs3)(CC1)OC2 C#CCC(CC#C)C(=O)N1CCOCC(NC(=O)C(F)(F)CN2CCOCC2)C1 C1(NC(c2ccc(OC)c(Cl)n2)=O)CN(C(=O)CP(C)(C)=O)CCC12CCC2 N1(C(c2c(F)ccc(C)n2)=O)CCC2(CCC(NC(=O)C(C)C3CCCO3)C2)C1 c1(C(=O)NCC(C)N(C)C(c2cc(N)c(Cl)c(O)n2)=O)cc(S(C)(=O)=O)co1 c1(CCCC(=O)N(CCOC)CCNC(C2CCOCC2)=O)ccc(F)c(F)c1 n1(CCC)nccc1C(=O)NCC1(C(=O)NCC2CCC2(F)F)CC1 N(C1CCc2ccc(Br)cc21)C(C1CCN(C(CC2N(C)C(=O)CC2)=O)CC1)=O c1(OC)ccc(Br)c(F)c1C(=O)NCC(=O)NC1CC(N(C)C)C1 C1(C#N)(OC)CC(C(=O)N(C)CCN(C(=O)CC2CCCCO2)C)C1 Cc1ccc(I)cc1C(N1CC(F)(F)CC1C(N1CCC(CF)CC1)=O)=O c1(C(=O)NC2CN(Cc3c(C)cc(C)[nH]3)CC2O)cc(C)ccc1C C1(C(=O)NC2C(C)(C)C(F)(F)C2)CC2CCCC2N1C(=O)CSC1CCCCO1 C1(NC(CC(CC)SC)=O)COC2(C1)CN(C(=O)C(C)(C)n1cncn1)C2 C(=O)(C(O)CCCNC(c1cccc(N)c1F)=O)N1CC(C)(CF)C1 CC(O)(CC(=O)NC1CN(C(C2CCC3(CC2)CC3)=O)CC12CC2)C(F)(F)F N(C1CCCn2ncnc21)C(C(=O)NCCCC1CCOCC1)=O CCCC(C(=O)NCC1CCCN1C(=O)Cc1sc(C2CCC2)nc1C)OC N(C(=NCCN1CCOCC1)NCC(C)(C)C)C1CC(C)OC1 c1(C(=O)NC(C)C(C)NC(c2cnc3c(c2)COC3)=O)nnn2c1CSCC2 CC1CCCC(C(N2CCN(C(c3ncnc(O)c3F)=O)CC2)=O)CC1 c1(C(=O)NC(CC)CNC(c2cnc(O)o2)=O)sc([N+](=O)[O-])cc1Cl C=C(Cl)CC(C(=O)NC1CC(C2CC2)C1)NC(=O)C1=CCCCO1 C(=O)(C1=Cc2ccccc2C1)NCCC1N(C(CN=S(C)(C)=O)=O)CCSC1 C1(CCNC(C(CNC(C)=O)F)=O)CCCN(C(=O)C(C)OC2CCOC2)C1 Cc1cc(C(=O)NC(C(=O)NC2CC2c2ccco2)C2CCCO2)cc(O)n1 c1(CN2CCCC(C(=O)Nc3cccc(OC)c3)C2)cccn2nnnc12 N1(C(C2C(C)C2)=O)CCCC(N(C(=O)COc2cn[nH]c2)C)C1 C1(C(=O)Nc2cncnc2)CCc2onc(C(=O)N3CC4(CC4)CO3)c2C1 C1(C(N(C2CCS(=O)(=O)C2)CC#C)=O)CCN(CC(N2CCCCC2C)=O)CC1 c1(C2(C(=O)Nc3cn(CC4(c5ccccc5)CC4)nn3)CCC2)ccc(Br)cc1 C(=O)(C(F)(F)CSc1ccc(F)cc1)N(CC(C)NC(c1cnc(C#N)s1)=O)C c1(C(N(CCCN(C(C2C(C)(C(=O)OCC)C2)=O)C)C)=O)cnc(C(F)(F)F)s1 c1(CC(N2CC3C(C2)N3C(c2ccc(F)c(O)c2)=O)=O)ccc(O)nc1Cl c1(C(=O)NCCC2CC(F)(F)CN2C(C23CC2C3)=O)c[nH]c2cccnc12 C(=O)(C1CCOc2ccccc21)C1CC(CCN=c2[nH]c(=N)[nH]c(=NCCC)[nH]2)C1 c1(C(=O)NCC2COCC2NC(=O)C(=Cc2ccccc2)F)cc([N+](=O)[O-])c[nH]1 C1(C(=O)NCC(C)(Cn2cccn2)NC(=O)CCC(C)(F)F)CC(C)(C)OC1(C)C C(=O)(CCC(C)CC(=O)NOC(C)(C)C)NC(CC(C)CN(C)C)=O c1(NC(C2CC(C)CN2C(C2CCCCO2)=O)=O)ccc2scnc2c1Br N1(C(C(CC)C)=O)CC2(CNC(c3conc3C)=O)CCC1CC2 c1(C(=O)NCC2(NC(CC3(C)CC3)=O)CCOC2)cnc2n1CCCC2 Cn1cncc1C(=O)NC(CNC(=O)CC1(CO)CC1)Cc1ccccc1 c1(CN2CCCC(C)(C(N3CCCOCC3)=O)C2)ccc2ccsc2c1 C1(NC(c2c(C)nc[nH]2)=O)CN(C(=O)Cn2ccnc2C(C)C)C2CC12 CC1CN(C(=O)C=Cc2ccn(C)c2)CCCN1C(C1CCC12CCC2)=O C1(O)(CC(=O)NC(C(=O)NCC(C)CO)c2cccs2)CCOC1 c1(N2CCN(C3C(OC)CCC3)CC2)ncnc2ccsc12 c1(CCC(=O)NCC(CNC(C2CCC(N(C)C)C2)=O)OC)ccc(F)cc1 N1(C(c2cnc(CC)o2)=O)CCC(NCC(=O)N(C(=O)C(C)(C)C)C2CC2)CC1 c1(OC(C)C(=O)NCC2CN(C(C3(Cl)CC3)=O)CCN2C)ccc(F)cc1Cl N(C1CCc2cc(F)c(F)cc21)C(N1CC(CC)N(C(=O)C2CC2)CC1)=O C(=O)(CC(C(C)C)OCC)NCC1(F)CCN(C(C=CC)=O)C1 c1(CC)ccc(C(N)C(N2CCC(C3CCCN3)C2)=O)cc1 Nc1cc(F)cnc1C(=O)NC(CC1(CO)CCC1)C(=O)NCC(O)CF Cn1c(=O)c2c(n(CC(=O)NC3CC(O)CN3C(C)(C)C)c1=O)CCC2 N1(C(c2c(N)c(Cl)ncc2)=O)CCN2CCOCC2(CNC(=O)CC2CCCO2)C1 c1(CC(=O)NC2CC(C)N(C(C3COCCN3C)=O)CC2)nc2ncccn2n1 CCCC(CC(=O)NCCc1cnn(CSC)c1)NC(=O)CC1COCC1O c1(OC)cccc(Cl)c1CC(N1CCC(O)(CNC(C2CC=CCO2)=O)C1)=O N1(C(c2csc(C)n2)=O)CC(C(=O)NC2(CCCC)CC2)OC(C)C1 c1(C(C)=O)cccc(C(N2CC(O)(CNC(C3(c4cccs4)CC3)=O)C2)=O)c1C C1(C)(C(=O)NCCC(C)NC(c2ccc(OC)o2)=O)CCC(=O)NC1 N1(C(C(c2ccco2)NC(C2CCC3(CCC3)C2)=O)=O)CC2CC2C2CC12 c1(-n2cc(CCCC)nn2)cccc(NCc2cc(Br)c(C)s2)c1 C1(C(=O)NCC2(CN(C(c3c(CC)scn3)=O)C)CC2)CCCN1N=O c1(C(N2C(C(C)C)CN(C(=O)C(C)(C)CF)CC2)=O)cccc2c1OCC2 c1(C(N(CC(C)N(C)C(c2cccc(C(C)(C)C)c2)=O)C)=O)ccc(N)c(Cl)c1 N1(C(CSC(C)(C)C)=O)CCN(C(=O)CC2CC3CCC2C3)C(C2CCCC2)C1 c1(OC)ccc2ccccc2c1CS(=O)C(c1ccc(O)c(C)c1)C C1(NC(C=C(CC)CC)=O)CC(CNC(=O)C(c2ccc(O)cc2)(C)C)C(O)C1 N1(C(C(=O)NC)CCC2CCCCC2)CCCCC12CCC2 C1(NC(C2(COC)CN(C(C3CCC3)=O)C2)=O)CC2(C1)CC(O)C2 C12(NC(CCCOCC)=O)CCCCCC1N(C(c1cnc(O)c(F)c1)=O)CC2 c1(C(=O)NCC(CNC(c2cc(C)n(CCO)n2)=O)(C)O)cccn2cnnc12 CCCCC(CC)CC(=O)NC1CCCC2CN(C(C3(C)CC(C#N)C3)=O)CC12 Cc1nn(C)c(N)c1C(N1CCC(C)C(CC(=O)NCC2CC3(CC3)C2)C1)=O N(C1CCc2ccccc21)C(c1ccc(C)c(C)c1F)c1nnnn1C c1(OC)cc(-c2cnc(NC(c3ncoc3C(F)(F)F)=O)s2)ccc1OC(C)=O C(=O)(C#CC1(C)CCCO1)N1C(C)(C)C(CC(=O)NCCOC(F)F)CC1 Cc1nc(C)c(CC(=O)NCC(C)CNC(=O)C=C2CCC(C)C2)c(O)n1 N1(C(CN(c2ccsc2)CC)=O)CC2CCC1CN2C(=O)CC1CC2(CC2)CO1 C1(C(=O)NC(C)C(C)(C)NC(=O)CCSC(F)(F)F)CN2CCN1CC2 N#Cc1cn[nH]c1C(=O)NC1CCN(C(C2CCCC3CC23)=O)C1 c1(N2CC(CCCCN(C(=O)CCCn3ccnc3)CCO)C2)cc(O)nc(O)n1 CCC(CN(C)C)C(=O)N1CCCC1CC(=O)N(C)Cc1cccc(O)n1 CC(C)CC(C(=O)N1CCC(CC(C)C)(C(F)(F)F)C1)N(C)C C1(C(N2CC3(CCCCC3)CC2CO)=O)CCc2ccccc2OC1C(F)(F)F C(=O)(CCCCCC(=O)NCC1(O)CC(NC(C2CC2NC(C)=O)=O)C1)NC C1(C(N(CCC#N)C(C)C)=O)CCN(C(=O)C(C)Oc2ccccc2C)CC1 N1(C(c2nc(C)c(C)o2)=O)CCCC(C)(C)C1CNC(c1cn[nH]c1)=O c1(C(N2C3CCN(C(=O)NC(C(=O)OC)C)C3CC2)=O)c(O)ccc2nc[nH]c12 c1(CN(C(C(C)OC(c2nn(C)cc2Br)=O)=O)C)ccc(F)cc1Br c1(CNC(C2N(C(C3CC3c3ccsc3)=O)CCC2)=O)cccc(OCO)c1 C12CN(CC1O)C2=O.c1(-c2n(C(C)(C)C)cnc2)ccc(NS(C)(=O)=O)cc1 c1(NC(=O)NC(C(C)C)C(F)(F)F)nnc2c(C(F)(F)F)cccn12 C=CC(CC)C(=O)N1CC=CC(C(=O)NCC2=NOCC2)C1 CCCC(CNC(=O)Cc1ccn(C)n1)C(=O)NOC1CCOC1 Cc1n[nH]c(C)c1CC(=O)NC(C)CC1CN(C(C2C=CC=CC=C2)=O)C1 C(=O)(C(O)C(CCC)NC(c1ccnc(O)c1)=O)NCCCCC#CC N1(C(C2CC(C)CN2Cc2sc(Br)nc2Br)=O)CCOC(C#N)C1 c1(CC(=O)NC(c2cc(C)cc(C)c2)CCO)cc(F)c(Cl)cc1[N+](=O)[O-] CC#CCCCC(=O)NCCn1cc(C(=O)NCCN(C(C)C)C(C)C)nn1 C(=O)(C1=C2CCCN=C2NN1)N1C(C2CCN(C(C(C)(C)CF)=O)C2)(C)C1.C1CC1 C1(NC(C(C(C)C)NC(c2cc(C)n(C)c2)=O)=O)CC(C)CC(C)C1 C1(C(=O)NC(CCCNC(C2CC(CC)C2)=O)c2ccccc2)CC(=O)N(C)C1 n1(CC)ncc(C(=O)N(C)CC2CCN(C(=O)COC3CCC3)C2)c1C C1(O)(CNC(C2CC(C)SCC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1 CC(C(=O)NCCCN(c1ccc([N+](=O)[O-])cc1)CC1CC1)C(C)S(C)(=O)=O CC(CF)C(=O)N(CC(C)(C)CNC(=O)C(C)Cc1ccco1)CCO C=Cc1cncc(C(N2CCCCC2CCCNC(C2CCCN2N=O)=O)=O)c1 CC1CCCN(C(C2COC(C)(C)C2)=O)C1CNC(c1c[nH][nH]c1=N)=O C1(C(=O)NC(CCC(C)C)=O)CCN(C(=O)CO)CC1F C1(NC(C23CC2CN(C(c2cnc(C4CC4)o2)=O)C3)=O)CCC12CCCC2 c1(C(=O)NCC2CN(Cc3cc(Cl)nc(Cl)c3)CCO2)cc2cc(F)ccc2s1 C(CC(CC)C(=O)NC(CC(C)C)C(=O)N1CCN(CC)C(C)C1)=CC C1(C(=O)NC2(CC=C)CN(C(=O)CC3CCCCCC3)C2)CCS(=O)(=O)N1 N1(C(Cc2c(C)nn(C)c2)=O)CC(C)CN(C(=O)C(C)(C)CCC#N)CC1C S(=O)(=O)(c1cnccc1N1CC=CC(O)C1)N(C)CC1(OC)CCOC1 C1(C(=O)NCC(c2ccc(C)cc2)N(C)C)OC2(CCNCC2)C(O)C1 Cc1ccc(C(=O)N(CCCC(=O)N(CCCC(C)(F)F)C)C)c(O)c1 N1(C(CC=C)=O)CCCCC1C1CCN(C(c2c(Br)cnn2CC)=O)CC1 C12(C(N3C(C(C)(C)C)CCCC3)=O)CCC(CC1)CO2 c1(N2CC3CC(NC(C4=C(C)CCCC4)=O)CC3C2)nc(Cl)nc2c1CCOC2 N1(C(CCN(CCCCOC)C)=O)CC(CNC(=O)C(O)CN(C)C)CC1(C)C C1(C(N2CC(F)(CC)C2)=O)CC(NC(=O)CN2CCCNC2=O)CCO1 N1(C(Cc2cn(CC)nc2)=O)CC(N(C(=O)CSCc2ccccc2)C)C(O)C1 N1(C(C(C)OC(C)=O)=O)CCOCC1C(=O)NCc1c[nH]nc1C(C)C c1(SC)ccc(C(=O)NC2(C)CCN(C(=O)Cn3cncc3C)C2)cc1 N1(C(C(C=C)OC)=O)CCCC(C2CN(C(c3cnnn3C=C)=O)C2)C1 N1(C(C(CC)C)=O)CCC(C)C1c1cn(-c2cccnc2Cl)nn1 c1(C(=O)NCC(C)C(=O)NC2CCn3cnnc3C2)ccc2cc[nH]c2n1 Cc1cc(OCC(=O)OCC(N2CC(Oc3cnc(F)nc3)C2)=O)cc(C)c1 C1(C(=O)NC(c2ccc(C)o2)CC)CC12CCN(Cc1cc(F)ccc1Cl)C2 Cc1ccc2c(C(N3CCC(N(C)C(C4CCC4(C)C)=O)CC3)=O)csc2c1 c1(C(=O)NCC2CCC(NC(c3cnc(C)n3C)=O)C2)ccc2cc[nH]c2n1 C(CCCCC(=O)N(CCNC(C1CC=CCC1)=O)CCOCCO)OCC C1(NC(C(C)OCCCCCC)=O)CCC12CCN(C(=O)CNC(C)=O)CC2 c1(NC(C)CNC(C2(O)CCSCC2)=O)ncnc2c1COC2 C1(CNC(C(CSC)O)=O)CN(C(C2(C)CCCC2)=O)CC(C)(C)C1 C(=O)(C1CCC(=O)c2ccccc21)N1C(CNC(c2[nH]cc(C)c2)=O)CCC1 C1(NC(c2c(CC)c[nH]c2)=O)CN(C(=O)C=Cc2cc(C)no2)CC1C CN1c2ccccc2N(CCNC(=O)NC2CCCC3(C2)N=N3)S1(=O)=O CC1CC(CNC(C2CC2C)=O)CCN1C(c1ccoc1)=O c1(OC)n[nH]c(C(N2CC(CCNC(C3(CF)CC3)=O)(OC)C2)=O)c1Cl CN(CCCC(=O)NC1CC(NC(C2CC(=O)NC(=O)N2)=O)CC1O)N=O C1(C)(NC(C2C(NC(C3C(OC)CC3)=O)CCO2)=O)CCCC1(F)F C1(C(=O)NC(CC#C)C(=O)OCC)(CC)CCN(C(c2cc(CC)sn2)=O)CC1 N1(C(C2(CSC)CC2)=O)CCN(C2CCCN(C(=O)C(C)O)C2)C(=O)C1 C1(CNC(c2cn(CCO)c(=O)nc2O)=O)CC2(CO1)CN(C(=O)C=CBr)C2 C1(COC)CN(C(c2csc(COC)c2)=O)CCN1C(=O)C=Cc1cnc[nH]1 C1(CNC(CCCC(=C)C)=O)CC(C)(C)CCC1NC(=O)C=Cc1cn(C)cn1 C1(C(=O)NCc2ccc(F)cc2)CC2C=CC1C2.O=C(CCCF)NC1CC(F)(CO)C1 C(=O)(C1=NNC(=O)C1)NC(CC(=O)N(CCOC)C1CC1)COC C(c1cnccn1)=CC(=O)NCC1OCCC1C(=O)NCC1(CO)CC1 C(CN=c1cc(CC2CC2)nc[nH]1)(c1nnn(C)n1)NC1CN(S(=O)(=O)C(F)F)C1 C12(NC(C(C3CCOCC3)C)=O)CC(CO)(C1)OC21CN(C(=O)OC(C)(C)C)C1 N1(C(CCC(=O)OC)=O)CCCC(NC(c2nccnc2C)=O)C(F)C1 N1(c2ncc(C)c(O)n2)CCC2(NC(=O)CCN3CCCS3(=O)=O)CCCC12 N1(C(C(CC=CCC)C)=O)CC2(CCC2)CC1C(=O)N(C)CCOC(C)=O N1(C(C(C)OCCCC)=O)CCCC(N(C(=O)Cc2ccns2)CC2CC2)C1 c1(OC)c(N2CCC(N(C(=O)C(C)OCC(C)C)C)CC2)ncnc1C N1(C(C(C)(C)SC)=O)CCCCC(C2CN(C(=O)C3=CCCOC3)C2)C1 C1(CNC(c2ccc(C(N)=O)o2)=O)CC(C(=O)NC2CC=CCC2)=NO1 CON(CCC(=O)O)C(=O)N1CCCC(COc2ccccc2)C1 c1(C(=O)NCC2OCC(C(=O)NCCC=CC)C2)ccc(F)c(O)c1 C1(CN(C(C2(SC)CC2)=O)C)CCN(C(=O)C(c2ccccc2)C)CC1O C1(CNC(c2c(CC)noc2C)=O)CN(C(=O)CNS(N)(=O)=O)CC(C)(C)O1 c1(C(=O)NCCCN(C(C)=O)CC)cn(CCOC)nn1.C1(=O)C(C)N1 N1(C(C(C)OCC=C)=O)CC(C2CCN(C(c3scc4c3OCCO4)=O)CC2)C1 N(C(=NCC1CCS(=O)(=O)C1)NC1CC1)CC(C)(C)C1CCC1 S(=O)(=O)(c1c[nH]c(CCC(=O)NCC2CCC(OC)(OCCCO)C2)c1)NC C1(NCc2ccc(C(=O)OC)o2)CS(=O)(=O)CC1NC(c1cccc(SC)n1)=O CN1CCN(C(=O)C(C)(C2CCC2)NC(=O)CN2CCOC2=O)CC1C1CC1 C(C(O)C(=O)NCC1CCCC1NC(=O)CCc1cnoc1)N(C)C c1(OC)cc(N=c2scc(-c3ccoc3C)n2-c2c[nH]nc2C)ccc1C(N)=O C1(C)(NC(CNS(C(C)CCN)(=O)=O)=O)C2CC3CC(C2)CC1C3 N1(C(C2ON=C(C)C2)=O)CC2CCCC1C2CNC(c1cc(C(C)C)[nH]n1)=O c1(C(=O)OC)cc(N(C)C(C2CCCCN2C)=O)ccc1C.CO c1(NC(C2C(NS(CC(=O)OC)(=O)=O)C2)=O)cc(F)ccc1Cl CCCCCCCC(=O)NCC1CCCN(C(=O)CCNC(C2CCC2)=O)CC1 C(=O)(C(C)(C)C(F)(F)F)N(C1CCN(C(c2cn(CC)nc2C)=O)CC1)CC Cc1noc2nc(C(N3CCCC(NC(C4(C(F)F)CC4(F)F)=O)C3)=O)ccc12 c1(C(=O)Nc2[nH]nc(C(C)NC(=O)OC(C)(C)C)n2)ccc(C)c2[nH]c(C)cc12 N1(C(=O)COc2ccccc2F)CC2CC1CN2C(C1CC2(CC2)CO1)=O CC1(C)CN(C(=O)COc2ccon2)CC1CNC(=O)CC1C=CCC1 CCCCC(CN(C(=O)CC1CCOC1)CC)NC(=O)CCc1c(C)noc1C C1(NC(CCNC(C(C)(C)C)=O)=O)CC2CCC(C1)N2C(C1CCCOCC1)=O C(=O)(CCS(N)(=O)=O)N1CC(CNC(C(C(C)C)n2ccnc2)=O)OCC1 N1(C(Cn2c(C(C)C)ncc2)=O)CCCC2(NC(c3ccccn3)=O)CC2C1 c1(C(=O)NC2CCN(CC(=O)NCCOCC=C)C2)ccnc(F)c1OC C1(F)(C(=O)NCC2C(CC(=O)NC(C=C)C3CC3)C2)CC(O)C1 C(=O)(CCP(C)(C)=O)NC1(C(=O)NCCC2CCCCC2)C(C)CCC1 N1(C(Cc2n(C)cnn2)=O)CCC(NC(=O)COc2cccnc2Cl)C(O)C1 CC(C)(C)C(C)(C)C(=O)N1CC2CC2(CNC(=O)C2=COCC2)C1 Cc1cc(C(F)(F)F)nc(CN(C(=O)CC2CCC3CC23)CCNC(=O)C2CC2)n1 n1(CC)ccc(C(=O)N(C(C)C(=O)N(CCC(N)=O)C)C)n1 c1(C(=O)NCCCCN(C(C2C(C)OCCC2)=O)C)cc2cnccc2cc1F C1(C(N2CCCC(CCNC(=O)COCP(C)(C)=O)C2)=O)(CC)CCC(O)CC1 c1(C(c2nnnn2C2CC2)NC(CCNC(C)=O)(C)C)c(C)cnn1COC c1(NC(c2cc(-c3cn(CC=CCO)nn3)cnc2O)=O)ccc(F)c(Br)c1 c1(Sc2n(CC)nnn2)cccnc1Cl.C1(CCCN)CC1(Cl)Cl c1(C(=O)NCCN(C(=O)CCCc2nc(C(C)C)no2)C(C)C)ncc[nH]c1=O C1(C(=O)NCC(C)(F)CNC(=O)CC2CCC2)CCn2nnnc2C1 CCCC(C(=O)NC1(CO)CN(C(=O)C(C)c2cc[nH]n2)C1)OCC C1(C(=O)NC2(c3cccc(Cl)c3)CC2)CCC(O)CN1C(=O)CCN1CCC1 c1(CCNC(CCOC(C)C)=O)cc(C(=O)NCC2CCC(C)C2)on1 c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C3CCC(=O)N3C)C)C2)ccc1C C1(NC(CCS(=O)(=O)NC)=O)CN(C(C2(C)CCCS2)=O)CC12CCOCC2 N1(C(c2n(C)ccc2)=O)CCCC2CN(C(C3(c4cccs4)CC3)=O)CCCC12 CC(C)C(F)(F)CC(=O)N1CC(NC(c2c(O)cccc2Cl)=O)C(C)C1 C#CC1CCC(C(=O)NC2CCN(Cc3cc(C(=O)NC)c(C)o3)C2C)CC1 c1(OCC)ccccc1C(N1CCCC(NC(=O)C(C)CF)C1)=O C1(N(C)C)CN(C(=O)CC2CC3(CC3)CO2)CC1CNC(=O)C(C)(C)CF C(C)(CO)(C(=O)NCc1ccc(Cl)nc1)NC(C(C)O)=O CCC(C)C(C)C(=O)N(CCCCNC(c1cc2n(c1)CCC2)=O)C C1(C(N2C(CNC(c3cc(C(C)C)no3)=O)CCC2)=O)C2(CCC2)C12CCC2 C1(N(CCCCCO)C(C2C3C(=O)OCC23Br)=O)CCS(=O)(=O)C1 CC(C)C(CNC(c1ccnnc1O)=O)C(=O)NC(C(F)F)C(C)(C)C c1(CNC23CC(C(=O)NCc4ccnc(Cl)c4Cl)(C2)C3)cc(Cl)c(Cl)cc1F CC(C)CCCC(=O)N(CC(O)CNC(C1CC2C(C1)C2(C)C)=O)C C=CCC(CC(F)F)C(=O)NC1CN(C(=O)COCCCOC)C2(CCOC2)C1 c1(C(=O)NC2CC(C)(NC(c3ccc(SC)o3)=O)C2)cc(C2(Cl)CC2)n(C)n1 C1(C(N2CCC(n3cnnn3)C2)=O)(OC)CCN(C(=O)CC2CCSC2)C1 C1(NC(c2c(C)c(Br)ccc2)=O)CC2CN(C(=O)CCN3C(=O)C=CC3=O)CC2C1 C1(C)(CC)CCN(C(C2CN(C(=O)C(CCN(C)C)N(C)C)CCO2)=O)C1 N1(C(C(COCC)C)=O)CCC2(CC1)CC(NC(=O)CC(C)CC(C)(C)C)C2 CC(C)C(C(=O)N1CCC(CN(C(=O)Cc2cocn2)C)CC1)NC(N)=O C#CC1(C(N2CC3C(NC(=O)CSc4nc[nH]n4)C3C2)=O)CCCC1 Cc1cc2[nH]c(C(N3CC(O)(CNC(C4CC5CCCC(C4)C5)=O)C3)=O)cc2o1 C1(NC(CCCC=C)=O)CN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC12CC2 c1(C(=O)NC(CC)CNC(C2(C)CCCO2)=O)cc(F)cc(Br)c1C C1(N(C(CC(CC)C)=O)C)CN(C(=O)CCCCN(C)C)CC1(C)C C=CCCCCCCC(=O)NC1C=CCCC1C(N1C(CO)CC1C)=O O(N(C(=O)CONC(=O)Cc1ccc(OC)cc1)C(C)C)CC c1(C(N(C2CN(C(C3(F)CCC(C)CC3)=O)CC2O)C)=O)cc2cc[nH]c2cn1 C1(C(=O)NC(C2(O)CN(C(CCOC(C)C)=O)C2)C)CCC(F)(F)CC1 N1(C(c2c(N)cn(C)n2)=O)CCCC(C)(CNC(=O)CCOc2cccnc2)C1 c1(C(=O)NCC2(O)CCCN(C(COC)=O)C2)cnc2cc(C)ccc2c1 C(CC(C)C(=O)N1CCC(NC(c2c[nH]nc2C2CCCCC2)=O)CC1)OC CC(C)CC(C)C(=O)NCC1CC(F)(F)CN1C(c1ccoc1C1CC1)=O C1(NC(c2cc(CC)no2)=O)C=CCC(C(=O)NC2CC2O)C1 C12(CNC(CC#N)=O)CCCC(CN1C(c1ccncc1F)=O)C2 c1(C(CC)C(=O)NC(C)(C)CN(C)C(C2(C)CC2(C)C)=O)ccc(OC)cc1 C(C(C(C)C(C)C)NC(=O)COCCN(C)C)NC(C1(CC(C)C)CCC1)=O Cc1[nH]nc(C(N2CCC(C)N(C(=O)Cc3ncn(C)c3C)CC2)=O)c1[N+](=O)[O-] N1(C(C(C=C)C)=O)CCC(CNC(=O)CSCC(F)(F)F)C(F)(F)CC1 Cc1ccc(C(=O)NCC2(F)CN(C(C3CC3C(C)(C)O)=O)C2)c(C2CC2)n1 C1(C(=O)NC(C#C)C)CCCN1C(=O)C=CC1CCCC1 C1(CNC(Cc2ccc(C)s2)=O)C2CN(C(=O)Cc3ccccc3)CC12 c1(C(=O)NCC#CCNC(C2(F)C(C)OCC2)=O)ccc2c(c1)OCCC2 c1(NC(C2(CCC)CC2)=O)cc(Cl)c(C(F)F)cc1F N1(C(C2CC(=O)NCC2)=O)CC2Oc3cccc(NC(=O)CSC(F)(F)F)c3C2C1 C(=O)(C1=COCCC1)N(C(CNC(C1CCC(NC(C)=O)CC1)=O)C)C1CC1 C1(CCNC(C(CC)O)=O)CCN(C(=O)CN2CC3CC3C2)CCC1(F)F N1(CCSc2cnc(CC(C)C)[nH]2)CN(C)C(=O)C1C C1(C(=O)NC(Cc2ncn(C)c2)C(=O)O)CCCC(C)(C)C1 c1(OC)ccc(C(=O)NC2CCC(CC(=O)NC(C)CO)C2)cc1 Cc1ccc(OCc2cn(CCNC(=O)NC3CCC(=O)CC3C)nn2)cc1C c1(C(=O)NC(Cc2ccccc2)CCO)cc(Br)cnc1Br c1(CC)cc(C(=O)NC2CCN(C(c3cn(C)nc3CC)=O)CC2C)c(C)nn1 N1(C(C2(NC(CC3C(CC)C3)=O)CCOCC2)=O)CCCCC(C)(C)C1 C1(CNC(C(COCC)NC(=O)CC2CCCC23CC3)=O)CC(=O)N(OC)C1 C=CC1(C(N2CC(O)(CC)C2)=O)CCN(C(=O)CC2C=CCC2)C1 CCC(CCOC)C(=O)N(CCN(C(=O)C(C)CSC(F)(F)F)C)C(C)C c1(C(=O)NC(C(C)C)CNC(=O)CC(C)(C)c2cccs2)cc(F)cc(N)c1F c1(C(=O)NCC2(C)N(C(C3C(COC)C3)=O)CCC2)cc(N)c(Cl)cn1 C1(C(=O)NC(c2cncnc2)C)C=CCCN1C(N1CCOCC1)=O N1(C(Cc2c(C)n(C)cn2)=O)CCC2(C1)CN(C(c1nnn3c1CCC3)=O)C2 C=C=C(C)CC(=O)NCC(C1CCN(C(C2(F)CC=CCC2)=O)CC1)F C(=O)(C(O)C(F)(F)F)N1CCC(CC(=O)N(C)CC2CC2C2CC2)C1 c1(C(N(C2CN(C(C3(OC)CCCOC3)=O)C2)C)=O)cnc(C(F)(F)F)cc1C Cc1c(Cl)c(C(N2CCN(C(c3cc(C4(C)CC4)n[nH]3)=O)C(CF)C2)=O)nn1C c1(CNC(C=CC(C)NC(=O)Cc2cccnc2)=O)cccc(C#N)n1 CC(CCNC(c1ccc(N2CCCC(O)C2)cc1)=O)CCC(=O)O C1(NC(CCn2c(C(C)C)ncc2)=O)CCCN(C(c2cc(Cl)no2)=O)CCC1 c1(CC(=O)NCC(CC=C)NC(c2ccc(SC)nc2)=O)c[nH]ccc1=O C1(NC(COCc2nnc(C)s2)=O)CCC2CN(c3ccc(C#N)nn3)CC2C1 Brc1ccc2nnc(COCC3CCCCC3Oc3ccccc3)n2c1 CCCC(C)CC(=O)NCC(C)(C1CC1)NC(=O)CSCc1nnc(C)n1C c1(C(=O)Nc2nccc(F)c2F)ccc2ccc(C3=CCNCC3)cc2c1 C1(F)(C(=O)NC2CC3CN(C(c4c(C)coc4)=O)C2C3)CS(=O)(=O)CC12CCC2 CC(=O)CCN=C(NCC(C)C)NC1CCC(C(N)=O)C1 CN1CCCCC(C(=O)N(C)CCNC(C2(c3ncco3)CCC2)=O)C1=O C1(CNC(c2c(F)cccc2F)=O)CN(C(c2ccccn2)=O)CC12CCC2 CC1(C)COC(C(N2CC3C(C(=O)Nc4cncc(Br)c4)C3C2)=O)C1 c1(CC(=O)N(C(=O)CN2CCCC(C(N)=O)C2)C)cccc(Cl)c1Cl.C(=O)(OC)N C1(NC(C)=O)CN(C(c2cccc(C)c2)=O)CC1C1CC1 C1(CNC(C2(CC=C)CCOC2)=O)CC2(CO1)CN(C(C1(CO)CCCC1)=O)C2 N1(C(C=CCCC)=O)C2CCC1CC(CNC(=O)C(c1cscn1)NC(C)=O)C2 C(=O)(CCCCN=[N+]=[N-])NCCC(CNC(=O)C(C)Oc1ccccc1)OC c1(C(N2C3CN(C(c4cccc(C)c4F)=O)CC2C3)=O)cc2ccccn2n1 N1(CCOC)CCC(c2nnnn2C2CCCC2)(NCC2CCCSCC2)C1 C=C(C(=O)NC1(CO)CN(C(c2cnc(O)cc2O)=O)C1)C(F)(F)F N1(CCNC(C2CC(NC(c3c(C)oc(C(C)(C)C)c3)=O)C2)=O)CCC(F)(F)CC1 C12(NC(CC(CC)O)=O)CCC(CN(C(=O)CC=CCc3ccccc3)C1)C2 C1(CC)C(C(N2CCC(O)CC2)=O)CCN1C(C1CCSCC1)=O N1(C(C(CC)CC)=O)CCN(C(=O)C(C)CC2CCC2)CC1c1ccccc1Cl N1(C(c2cc(C#C)cc(Br)c2)=O)CCOC2(C1)CN(C(C1CC1CF)=O)C2 N(C1c2ccccc2CC1(F)Cl)C(=O)CSc1ccc(Br)cn1 C(CCC(C(=O)N1CCCC(CCF)C1)NC(c1cccn1C)=O)OC N1(C(COCP(C)(C)=O)=O)CC(NC(=O)CNC=O)CC12CCC2 C1(NC(c2nc(C)n(C)n2)=O)CCCCC12CCCN(C(=O)CC(C)F)C2 CC(CN(C)C)CC(=O)N(C)CCC1CCN(C(=O)C(F)(F)C2CCCC2)CC1 CCCCCC(C)CC(=O)N(CCC)CCNC(=O)CCn1cccn1 CC(=NO)C1CC(C(=O)NCC(C(C)C)NC(C2(C(F)F)CC2)=O)C1(C)C c1(C(=O)NC(c2cc[nH]n2)C)ccc(CNC(c2cnsc2)=O)nc1 c1(N2CCC(c3ccc(Br)cc3)(C(=O)OC)C2)cc(C)nc2ccnn12 CC1(CNC(c2cncc(F)c2)=O)CCN(C(c2nn[nH]c2Cl)=O)C1 C(CCNC(=O)C1CC1)(C(C)C)NC(CN(C(C)=O)C)=O c1(C(=O)Nc2cc(C(=O)OC)ncc2Br)cnc2onc(C)c2c1 c1(C(=O)Oc2c(C)ccc(C)c2)c2c(nn1C)CCN(C(=O)CCC(C)C)C2 N1(C(C(=O)N(C(C)C)C)C)CCCCC(NC(c2ccc(=O)n(C(C)C)c2)=O)C1 C1(NC(C2CC(=O)N2)=O)CC2CCC1CN(C(c1cc(C(C)(C)C)sc1)=O)C2 N1(CC(CC)CC)CCC(CC(=O)NCCNC(=O)CCCF)CC1 C=CCC(CNC(C1CCCCC1)=O)C(=O)N(C(C)C(C)(C)C)C CN1CC(NC(N2CCCC2CN)=O)CC12CCC2.c1(O)ccc(C#N)cc1 N1(C(c2cccc(OC)c2)=O)CC2(CCCC2NC(=O)C(C)CC2CCC2)C1 N1(C(COC2CCN(C(Cc3c(C)cnn3C)=O)C2)=O)CC2(OC)CCC1CC2 c1(C(N2C(C)(COC)CC2)=O)cc2c(Br)cccn2n1 C(CCCC(=O)N(C)CC=CC(=O)N(C)Cc1occc1C)OC C1(CNC(C(C(=O)OCC)F)=O)CC2CCC(C1)N2C(=O)C(C1CCOCC1)O C1(C(N2CC(NC(CCc3c(C)noc3C)=O)(CO)C2)=O)OCC2CCCC12 n1(C2N(CC3CN(C(c4cnn(CC)c4C)=O)C3)CCC2)cc([Si](C)(C)C)cn1 C(=O)(C(C)N=[N+]=[N-])N(CC(=O)NCC=C=C)CCOC c1(C(=O)NC2CC3CN(C(C4(COC)CC4)=O)CC3C2)coc2cc(C)ccc12 Cc1ccc(C(CC(=O)O)NC(c2cncn2-c2cccc(F)c2)=O)cc1 CCC(C)(C)C(O)C(=O)NC1CC2(C1)CC(CNC(=O)CCc1nccs1)C2 c1(C(=O)NC(C)CC(C)NC(=O)C=Cc2c[nH]c(=N)[nH]2)cccn(C)c1=O c1(CC)nnsc1C(N1CCC1CNC(=O)CC1CCNC1=O)=O c1(CC)ccc(N)c(C(=O)NCCCCNC(C2CC3(CC3)CN2C)=O)c1 CCC(C)C(C)NS(=O)(=O)CC1CN(C(=O)OC(C)(C)C)C1 N1(C(C2(C(=O)OCC)CC2)=O)CCC(N)CC1.C(=O)(C(C(C)C)OC)C(=O)C(C)SC c1(N(C)C)ncc(C(=O)NC2CC2CNC(=O)CCNC(c2ccco2)=O)cc1Cl c1(C(N2CC(CC)C(C(=O)NC3CCN(CC)C3)C2)=O)nc(C)ccc1C C=CC1(C(=O)NCCC2(C)CCN(C(c3coc(C(F)(F)F)c3)=O)C2)CCCC1 CC(C)C(C(C)NC(C1(F)CCCCC1)=O)NC(c1coc(CO)c1)=O c1(CN(CCCNC(Cc2c(C)noc2)=O)C(C)C)cc(Cl)ccc1Br CCCCC(O)C(C)C(=O)NC1CCC(CC(=O)NC2CC=C(C(C)C)CC2)C1 C(=O)(CCCCC(N)=O)N1CCC=C(CNC(c2c(C)ccnn2)=O)C1 C1(C(=O)NC(c2cc(C)nnc2C)=O)COCCN(CC)C1.C1(=O)NCCN1 CC1=CCCN(C(=NCc2ccc(N(C)C)cc2)NCC(c2cccs2)O)C1 N1(C(=O)NCC(c2cccc(I)c2)C)CCCC(C)(O)C1 N1(C(c2cc(C)n(C(C)C)n2)=O)CCCC(O)(c2cn(C3CCOC3)nn2)CC1 N1(C(c2ccc(C)nc2O)=O)CCCC2(CCCN2C(C2COCCN2C)=O)C1 Cc1ccnn1CC(N1CCC(NC(C2(CCOc3ccccc3)CC2)=O)C1)=O C(CC(=O)NC1CN(C(C)C)C1)(C(F)(F)F)NC(CCC)=O CCC(C(=O)N1CC(O)(CCNC(C2CC2Cl)=O)C1)NC(C)=O C1(NC(C=CC=CC)=O)C2CC3CN(C(=O)COC)C1C3C2.C1(OCC)CCCCC1C C1(NC(C(C)SCCCC)=O)CCCCC1CNC(=O)C(C)C1CCC1 C1(NC(c2ccc(CCC=C)cc2)=O)(CO)CCCN(C(C2CC2C2CC2)=O)C1 O=C1CCN(C2CN(C(c3c[nH]nc3Br)=O)C2)C(=O)N1 CC(O)CCCCCC(=O)NC(C)CNC(=O)CCC1(C)CC1 C1(C(=O)NCC(CN(C(=O)Cn2cc(CC)cn2)CC)(C)C)CCC2CC2CC1 CC1CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1C(=O)NC1CCOCC1F Cc1[nH]c2ccc(Br)cc2c1CC(N1CCCCC(c2ccc(F)cc2)C1)=O Cc1cc(F)ccc1C(O)C(=O)NCCN(C(=O)Cc1ccco1)C1CC1 n1(CC(=O)N(C2CN(C(=O)C(C)(Cl)Cl)CC2F)C)ccc([N+](=O)[O-])n1 C1(C(=O)NCCC(C)O)CC(O)C(O)CC1C(=O)NC1(C)CCCCC1(C)C CC(=O)CC(C)(C)C(=O)NCc1cnn(C)c1C(N1CCC(N2CCCC2)C1)=O CC(C(=O)NOC1CCC1)C1CCN(NC(=O)CN2CCCCC2=O)CC1 N1(C(C2(CCNC(C(C(C)C)F)=O)CC2)=O)CCn2ccnc21 CC1CCNCCC1N(C(=O)CC1(O)CCC1)Cc1ccn(C)n1 C(=O)(C(C(C)(C)C)N(C)C(C)=O)NCC(C)(C)OCC1C(C(=O)OC)C1 Cc1cn(C)nc1C(=O)N(CC(=O)NC1CC(C(N)=O)C1)C1CCC1 c1(C(N(CCN(CCNC(C(CC)O)=O)C)C)=O)cccc2c1CCC2 C1(CNC(c2c(C)nc(C)o2)=O)CN(C(C23C(=O)C4CC2C3C4)=O)CC12CCC2 CC(C)C(CCN(C)C(C1CCC(F)C1)=O)NC(=O)CSC1CC1 N1(C(CC)C(N)=O)CC2CCC(NC(c3cc4n(n3)CCCC4)=O)CC2C1 CC1=C(C(=O)N2CCC(N(C)C(C3CCc4c[nH]nc4C3)=O)C2)CCCO1 CCCC(C)(CCC)C(=O)NC1C=CCC(C(=O)NOCCCCC2CC2)C1 c1(CC)cnc(Cl)[nH]c1=NCc1cc(O)nc(NC(c2cccc(OC)c2)=O)n1 N1(C(C2(C)CCC2)=O)Cc2nccn2CC(NC(=O)C(C2CCCO2)C2CC2)C1 C1(C(C)NC(N)=O)CCCN1C(=O)C(C1CCCCC1)C CC1(C)CCC(C)(C(N2CC3CCC3(NC(c3csc(C(F)F)n3)=O)C2)=O)CC1 N1(C(C=CC=CC)=O)CCOC(C)(CNC(=O)C(C)Oc2ccc(Cl)cc2C)C1 Cc1cc(C(N2CCN(C(c3ocnc3C)=O)CC2CF)=O)c(Br)c(C)c1 c1(OC)cc(C(=O)NCC2CC2CNC(=O)CCCC#N)nc(Br)c1 C1(NC(Cn2c(C)cc(=O)cc2)=O)CCN(C(c2cnccn2)=O)CCC1CO Cc1ccc(C(=O)NCC2CN(C(c3c[nH]nc3F)=O)CC2O)c2ccccc12 c1(C(C)NC(C2C(C(=O)O)CC2(C)C)=O)cccc(C(F)(F)F)c1F CN1N=C(C(=O)NC23CC(C2)N(C(=O)CC2CCCNC2=O)C3)CCC1=O c1(C(=O)NC(CNC(CCCOC)=O)CC(C)C)cc2nc(C)cc(C)n2n1 c1(CNC(C2N(C(C3N(C)CCOC3)=O)CCC2)=O)ccc(F)cc1F c1(CC)cccc(F)c1C(=O)N(C1CCN(C(=O)C(=O)C(C)(C)C)C1)C Cn1nc(CNC(c2ccccc2C#N)=O)c2c1CCN(C(=O)CC(C)(C)F)C2 C1(OC)CC2CN(C(=O)CN(C)C(C)=O)CC12.c1(CC(=O)N)cc2occc2[nH]1 c1(C(=O)NCCCC(C)NC(=O)CCc2cccc(O)n2)csc2cncn12 c1(C(=O)NCc2cc(C3C(C)C3)n[nH]2)cc2ccc(Cl)cc2o1 c1(C(=O)NCCC2N(C(C(CC)CC)=O)CCC2)cccc2cncn12 O=C1CC(CC2CCCCN2C(=O)CCN2CCCC(N3CCC3)C2)C(=O)N1 N1(C(c2c(CC)ncs2)=O)CCCCC(CNC(=O)Cc2conc2C)C1 C1(CNC(Cc2ncc(C)s2)=O)CC2COCC2N1C(=O)Cn1ncnn1 C=C(CNC(=O)C(C)(F)c1ccccc1)CCNC(=O)Cc1csc(CC)n1 N1(C(c2cc(CC)c(F)cc2)=O)CCC2CCC(C1)N2C(=O)Cc1ccoc1 CC1(C)CC(CNC(=O)C2=NOCC2)CN1C(=O)CC1(C(F)F)CC1 c1(N2CC(NC(CCC(=O)N(C)C)=O)CC(C)(C)C2)nccc(S(C)(=O)=O)n1 Cc1c(NCc2cccnn2)ncnc1N1CCCC(c2nncn2C)C1 c1(C(N(C(C)CNC(c2cncc(C)n2)=O)C)=O)cc([N+](=O)[O-])ccc1NC N1(C(C23CC(OC)C2C3)=O)CCN(C(c2cnc(N)c(N)c2)=O)CC1CO N1(C(CC(COC)(C)O)=O)CC2CCC1C1CN(C(=O)Cc3nc(C)no3)CC21 C1(CNC(C2CCC(C)(C)C2)=O)COCCN(C(c2ccccc2O)=O)C1 n1(CC)nc(C)c(CC(N2CC(O)CC2C(=O)NCc2cccc(Br)n2)=O)c1C N1(C(c2c(Cl)cn(C)n2)=O)CCC2CN(C(=O)CCc3cc(Cl)no3)CCC12 C1(CC)CN(C(=O)C(c2c(F)cccc2F)C)CCC1NC(c1[nH]cnc1C)=O CC1CC(NC(=O)CC2CCC(=O)O2)CN(C(c2cc(C3CC3)nc(O)c2)=O)C1 N1(C(C(c2cccnc2)OC)=O)CCC(NC(c2cc(Cl)no2)=O)CC1C C(=O)(C(F)(F)C(F)(F)C(F)F)NC1C(CNC(=O)CC2CCOCC2)CC1 C(=O)(C(C)(C)N=[N+]=[N-])NC(c1ccccc1)C(=O)NCC1CCC(C)CC1 C(=O)(C(O)Cc1ccccc1)O.c1(O)ccccc1.C1C(=O)CCC=CCCN1C C1(C)(CC(N2CC(O)(CN(C(=O)CCC3CCCO3)C)C2)=O)CC(F)(F)C1 C1(C(N2CCC(C(CO)NC(C3(CF)CC3)=O)CC2)=O)CN2CCN1CC2 c1(Nc2n(CCOC)c(N3CCC(F)(F)C3)nn2)ccc(Cl)c(F)c1 n1(CC(=O)NCC2C(NC(C(CCC)CC)=O)CCC2)cc(C#N)c(O)nc1=O C12(CNC(COC)=O)CCCC1N(C(c1cc([N+](=O)[O-])ccc1O)=O)CCC2 N1(C(C(C)C)=O)CCC(C2CC2)C1CNC(c1ccc(N2CCCC2)c(F)c1)=O C(=O)(CCCCC(=O)NCC1C(C)CCN1C(c1ccc(C)n(C)c1=O)=O)NC S(=O)(=O)(c1ccc2nc(N(C)C)sc2c1)NCCC(CNC(C1CC(=C)C1)=O)C C1(C)(CNC(C2(CCC)CCNC2=O)=O)CCCC1NC(=O)CCCCN(C)C c1(-c2n(-c3cccc(OC)c3)nc(CC(N)=O)n2)ccc2c(O)nnc(O)c2c1 C(N=c1nc(O)c2cccc(Br)c2[nH]1)c1cccc(CNC(C)=O)c1 NS(=O)(=O)c1cc(C(=O)NC2CN(C(=O)C=CC3CCOC3)CC2C2CC2)co1 N1(C(C(CCCC)N)=O)CCc2cc(Br)cc(F)c21 C(=O)(C(C)(O)C(C)c1ccccc1)NCCOCCNC(Cc1c(C)scc1)=O N1(C(c2cc(CC)nn2C)=O)CCC(C2CC2)(CNC(C2CCCOC2C)=O)C1 c1(-c2nccc(C(=O)OC(=O)CC3CCCCO3)c2)c(Cl)cccc1Cl N1(C(c2c(C(C)NC(c3ccc(F)cn3)=O)noc2)=O)CCC2CCCC2CC1 C(=O)(C1CCCc2ncnn21)N1CC(C)C(NC(=O)CCCN2CCC2)C(C)C1 c1(NC(c2cccc(-c3ncc4n3CCCC4)n2)=O)ccc2c(c1)CCNC2 c1(NC2CCC(SC)C2)ncc2c(n1)CCNC2 c1(CC)c(C(=O)NC2CCN(C(c3ccccc3SC)=O)C2(C)C)cccc1C C1(F)(CNC(CN2CC(C)C2)=O)CCN(C(=O)C(C)c2cccs2)C1 C1(CN(C)CC2CCN(C(c3cncc(Br)c3)=O)CC2)CCCC2(CC2)C1 c1(SC)ccc(C=CC(N2CC(F)(CNC(C3CC4CCC3O4)=O)C2)=O)s1 S(=O)(=O)(c1ccc(C(N2CC(NC(C3CCC3(C)C)=O)C(O)C2)=O)s1)NC C(CC(C)(CC)NC(C12CCC(C1)C2)=O)NC(C(C)OCC#C)=O c1(C(N2CC=CC(NC(C3(CO)CC3)=O)C2)=O)cc2c(=O)cc[nH]c2s1 n1(CCC)cc(C(=O)NCCC2CCC(NC(=O)CNC(=O)C3CC3)C2)c(C)n1 C(C1CCCCC1)=CC(=O)NCCCCN(C(=O)Cc1ccnn1C)C c1(OC)ccc(Br)c(CNC2CCCC(C(N3CCC(F)(CO)CC3)=O)C2)c1O C(=O)(CC(CNC(=O)CSCC(F)F)C1CCC1)N(C)CC1CCN(C)C1 c1(C(=O)NCC2CCCCN2C(C2CC3CC3C2)=O)cnc2c(c1)COCC2 C(C(C)(CC)C(=O)NC1(COC)CC1)NC(C(CN(CC)CC)F)=O C1(CNOCC)CCC(C2CC2)N1C(=O)C(C)COc1ccccc1 c1(CC)oc2ccccc2c1C(=O)NC1CC1CNC(c1snc(O)c1Cl)=O S(=O)(=O)(c1ccc(Cl)s1)NC1(CNC(C(CCOC)N(C)C)=O)CC1 c1(C(N(CC(C)CNC(c2cc(Br)c[nH]2)=O)C)=O)cc(Cl)ncc1Cl CC1CCN(C(C2CCC3(CC3)N2C(=O)C(O)CN2CCCC2)=O)CC1(C)C C(=O)(C(C(C)(C)C)OC)N(CC(C)N(C(c1cnc(C(=O)OC)s1)=O)C)C C(CC(=O)N(CCC(=O)N(C)C)CC(O)CO)=CC=C N1(C(CC2(C)N(C(CCC#CC)=O)CC2)=O)CCc2ccc(O)cc21 C1(NC(CCc2cnn(C)n2)=O)CN(C(C2COC3COCC23)=O)CC(C)(C)C1 c1(-n2c(C(CCCC)NCC=CC3CC3)nnn2)ccccc1Cl.SC c1(C(=O)NC2C3CN(C(c4c(SC)ccs4)=O)C(C3)C2)c(C)cc(C)nc1C CCC(CC)CCC(=O)N1CC(CF)(CNC(=O)COCC2CCOC2)C1 c1(-c2cc(C(=O)Nc3ncc(C#C)nc3)c(F)nc2)ccc2ccn(C)c2c1 CCC(C)C(C)CNC(=O)C(C)(C1CC1)N(C)C(c1ncccc1Cl)=O C1(C(=O)NCCCC(=O)Nc2cnn(C)c2)(CC)CCCCO1 CC1(C)CC(CNC(C2CCCO2)=O)CN1C(c1cc(C(F)(F)F)on1)=O C1(CNC(=O)OC(C)(C)C)CCC(NC(c2n[nH]c(=N)[nH]2)=O)C1 C1(C(F)F)(CO)CCCSC1.C1(C(N2CC3(C2)COCC(=O)N3)=O)CC(F)(F)C1 C(C)(C)(C(=O)N1CCC(OCCNC(=O)CSc2ccoc2)C1)N(C)C c1(C(=O)NC2CN(C(=O)C=CCF)C3(CCOC3)C2)ccc2ncccc2c1Cl c1(-n2ncc(C)c2)cccc(C(=O)NC(C)CC2CN(C(=O)CSC(F)F)C2)c1 C1(C(=O)NCCCN(C2CCCC2)C(=O)CN(C)C(C)C)CC1(C)C(F)F.CO C1(CNC(CCNC(=O)OC)=O)CC12CCN(C(=O)CC1CC13CC3)CC2 C(CCCCC(=O)N1CC(C#N)C1)NC(c1c(CC)ccs1)=O N1(C(c2c(C)ccc(O)c2)=O)C2CC(F)C(C2)C1C(=O)NC(c1ccn(C)n1)C C#CCCCC(C)C(=O)NCC(C)(C)C#CC(=O)NCC1=CCCOC1 c1(C(=O)NC2(C)CCCN(C(CC3(C)CCOCC3)=O)C2)cnc2c(c1)COC2 c1(C(=O)NC(C2CN(c3c(C#N)c(C)cc(C)n3)C2)C)ccc2ccccc2n1 N1(C(c2cnccc2Br)=O)CCC2(CCCN2C(=O)C=C2CCCCC2)C1 Cc1cnc(N2CCN(S(=O)(=O)N(C)C)CC2)c(S(=O)(=O)NCC(C)C(F)F)c1 c1(C(=O)NC2CN(C(CN(CC)CC)=O)C2)ccc(SC(F)(F)F)[nH]1 Cc1cc(C(=O)NC2CC(CNC(c3ccc(C#N)n3C)=O)C2(C)C)ccc1F CC(C)(O)C#CC(=O)NC1CC(CNC(=O)CCC2CCC(C(F)(F)F)CC2)C1 CC1CC=CCC1C(N1CCCCC1C1CCN(C(c2cc(Cl)cn2C)=O)C1)=O c1(CCC)cc(C(=O)NCC2CC(CNC(=O)C(C3CCOCC3)F)C2)c(C)o1 C1(CNC(CCn2ccc(C)n2)=O)CC2(CN2C(c2cc(C)on2)=O)CO1 CCCS(=O)(=O)C(C)C(=O)N1CC(c2cn(CCN(C)C)nn2)C2(COC2)C1 c1(C(N2C(C(C)(C)C(=O)NCC3CCCCC3)CC2)=O)c[nH]c2ncccc12 C1(C(=O)NCCC2CC(NC(C3N(C)CCC3)=O)C2)OCCCC1(C)C N1(C(c2ccncc2N2CCOCC2)=O)CC2(CCN2C(=O)Cc2cnccn2)C1 CN(C)S(=O)(=O)N(C)CC(N1CCC(N(CCO)C(C2CCCC(=O)O2)=O)C1)=O c1(C(=O)NC(CCCC)CC)cccc(S(=O)(=O)NCc2ccc(OC)cc2)c1 c1(NC(CNC(C(C)OCCOC)=O)C(C)(C)C)ncc(C2CC2)cc1C N1(C(C(CCCC)=O)=O)C2CCC1CC(NC(c1ncc[nH]c1=O)=O)C2 Cc1cc(C(=O)NCC2COC(CNC(=O)Cc3cccc(Cl)c3)C2)c(C)n1C C(C(C)(C)CC(=O)NOCC1CCOC1)NC(c1nc(C)sc1C)=O c1(CC(=O)NC(c2sccc2C(F)F)=O)ccccc1F.C12C3CN(CC13)C2 c1(C(=O)NC2CC(CNC(CCNC(C)=O)=O)C2)cccc(C)c1O N1(C(C(CC)O)=O)CCCC(O)(CN(C)C(c2cn(C)nc2C(C)(F)F)=O)C1 CN1CCCCC(C(N2CCC(C)(CNC(C3(C)CNC(=O)C3)=O)C2)=O)C1=O C(=O)(C#CC1(C)COC1)NCC1N(C(Cc2c(C)con2)=O)CCCC1C CC1CCC(NC(c2cc(N)c(F)cn2)=O)CN1C(c1cnc(C2CC2)s1)=O N1(C(C(N2C3CC(NC(C4(C)CC4Br)=O)CC2CC3)=O)=O)Cc2ccccc2C1 C=CCC(C(=O)NCCC1CCN(C(=O)Cc2csnc2C)C1)NC(C)=O C12(NC(c3cc(C)ncn3)=O)CCCCC1CN(C(C1CC1C1CCCC1)=O)C2 C1(C(N2C(C)CC(OC)C2)=O)CC2(CCN1C(C1CC3CCC1CC3)=O)CC2 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC(C(=O)NC2CCN(C)C2=O)CC1 CC(C)(C)C(O)CONC(c1ccoc1CNC(C1CCNC1=O)=O)=O N1(C(c2sc(C)c(Br)c2)C(=O)Nc2ccccc2)CCCCC(F)(F)C1 c1(CS(=O)(=O)N(CCC)Cc2cnn(C)c2C#N)ccc(Cl)cc1F C(=O)(C#CC1CCCCO1)C(=O)Cc1ccc(C(F)(F)F)cc1.N(CCN)(CC)CC c1(C(N2C(CNC(c3n(C(C)C)cnc3)=O)COCC2)=O)cc2n(n1)CCCO2 C#CC1(C(=O)NC(CCO)C(C)(C)O)CCN(C(=O)C=Cc2ccsc2)C1 C1(CN)CC2CCC1N(C(C1CCCN1C1CC1)=O)C2.C12(CCCCC1)C(=O)N2 CN1CC(NC(C2CCOC(=O)C2)=O)C(C(F)(F)F)C1 C1(CNC(COCCC#C)=O)CCN(C(c2nnc(S)n2C)=O)CC1O C(=O)(C1CCc2cc(F)ccc21)NCC(=C)CCNC(=O)C(F)(F)C1CC1 C1(NC(CC=C)=O)CCN(CCNC(c2csc(-c3ccc(F)cc3)n2)=O)CC1 C1(C(N2C(CNC(CC(C)Cc3ccc(Cl)cc3)=O)CC2)=O)CC2CCC1CC2 C1(NC(=O)C(O)CNC(C2(O)CCOC2)=O)CC2C=CC1C2 N1(C(c2ccc(C)c(Cl)c2)=O)CCC2CN(C(=O)C(C)(C)CN(C)C)CC12 CC1(CC(=O)NCC(Cl)NC(=O)CCCNC(=N)N)CC(F)(F)C1 Cc1cc(=NCC(O)c2ccc(Cl)c(F)c2)[nH]c(N(CC(C)CO)C)n1 CC1(C)CCC(C(=O)NC2CCCCC2CC(N2CC(OC(=O)C3CC3)C2)=O)C1 Cc1sc(=O)n(C(=O)N(C2CN(c3ncnc(C(C)(C)C)n3)C2)C)c1C c1(SC)ccccc1OCC(O)C(N1CCOC(CCNC(=O)C=CCF)C1)=O n1(CC)cc(C(=O)NC(C)(CO)C(=O)NCCSC)c(C)n1 C1(CNC(COCC#C)=O)(NC(C2CCCC2O)=O)CC2CCC1CC2 c1(C(N2CCN(C3CN(C(C(=O)NCC)=O)C3)CC2)=O)nccc(OC)c1OC c1(C(=O)NC(C)CC2CN(C(C3CCCC34CC4)=O)C2)cccc2c1OCCO2 CCC(C)(C#N)C(=O)NOCC(=O)NC1CCn2nnnc2C1 C(C)(C(C(=O)NCC)NC(C)=O)CC.C1(O)CN(C(=O)CC2(COC)CC2)CC1CC C(=O)(C(C)(F)C(=O)N(CC(O)C(=O)NCC(N1CCCC1)C)C)OC C1(C(=O)NCC(C)CN(C)C(c2c[nH]nc2-c2cccs2)=O)CCCN1C=O N1(C(C)C)CCCCC1C(N1CCCC1C1(NC(=O)C2=CCSC2)CC1)=O c1(CC)cnc(C(N2C3CN(C(c4cccnc4OC)=O)CC23)=O)nc1 C(CO)(C(C)N=c1[nH]c(=NC2CC(F)(F)C2)[nH]c2c(F)cc(F)cc12)SC S(=O)(=O)(c1cc(C)cnc1NCCCCCCN(C)C)N1CCCC(C=C)C1.S(C)(=O)(=O)N C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1CC(C)N(C(c2cc3n(n2)CCCO3)=O)C1 Cc1cccnc1CCC(=O)NCCSCC(N1CC(O)C(O)C1)=O c1(CC(=O)NC2CC(C(C)NC(Cn3ccc(C)n3)=O)C2)cccc(F)c1 CC1C(=O)N(CC(=O)N(C)Cc2cccc(CNC(=O)C=CCO)c2)C(=O)C1C C12(CNC(c3cncc(C)c3)=O)CCC(CN1C(c1cccc(=O)n1C)=O)C2 C(CC(O)CC(=O)N1CC(F)CC1CN(C(=O)CCc1ccccn1)C)SC c1(CN(C(C2C(C(C)NC(C=C)=O)C2)=O)CC)cccc(O)c1 C(=O)(CCCCN(C)C)NC1CC(CNC(CN(C)C)=O)C1 C=CC1(C(=O)NCCOCCCNC(=O)C(O)C(=O)OC)CCOCC1 C1(C(=O)NC(C(=O)OC)C2CC2)CCCCN1Cc1csc(NC(C)=O)n1 CC1CC2CN(C1)C(=O)CNC2=O.c1(NC(=O)OC(C)(C)C)cc(F)cc(Cl)c1 Cn1nccc1C(=O)NCCC1CCCN1c1nnc(CO)s1 Cc1ncc2c(n1)CCC(NC(CC(N)=O)C1CC1)C2.c1(N)nccc(N(C)C)n1 C1(OC(C)C(=O)NC2CCC2NC(c2nc(Cl)cs2)=O)CCCCCC1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CC2CN(C(c3cc(CO)c(C)o3)=O)CC2C1 C1(CNC(CC=C(C)C)=O)CCN(C(=O)CCCCOc2ccccc2)C12CC2 Cc1cc(NC(=O)CC2CC2(C)C)ccc1NC(C1CCC(O)CC1)=O C1(C(N(C2CCN(C(c3n(CC#C)ccc3)=O)C2)CC)=O)CC2(C1)CC2F c1(CNC(C2N(C(c3n[nH]c(C)c3C)=O)CCCC2)=O)ccc2c(c1)CCO2 C(=O)(CCCN(C)N=O)NC(CN(C(c1ccc(=O)n(C2CC2)c1)=O)CC)C C1(C(N(C)CC2CCN(C(c3snc(O)c3Cl)=O)C2)=O)CC2CCCC(C1)C2 C1(C(c2nnnn2CCN2CCOCC2)NC2C(O)CCC2)C2CC=CCC12 c1(C(NOC(C(=O)OC)C)=O)cncc(CNC(=O)C=CCF)c1 Cc1coc(C(=O)NC2CCN(C(=O)CC3(C)CC3)C2)c1C C1(NC(c2c(Cl)cc(C)s2)=O)CCN(C(=O)CCc2ccc[nH]2)C(C)C1 C1(N(C)C)CN(C(C2CC(F)CN2C(c2ccc(O)c(F)c2)=O)=O)CC12CC2 C1(C(N2C(CNC(c3c(CC)con3)=O)CC(O)C2)=O)Cc2nncn2C1 Cc1nc(SC(F)(F)F)sc1CC(=O)NCCNC(=O)CSC(F)F c1(SCCC(=O)NCC2CC(NC(=O)CCC3CCC3)C2)ccc(Cl)cc1 Cc1ccccc1C(C)CC(=O)NCCC(C(C)C)NC(=O)CN(C1CCC1)C C1(C(=O)NCC(CC)C)CC2CCC(C1)N2C(=O)CCCC#N c1(C(=O)OC)c(C)cc(C)c(NC(=O)Nc2[nH]c3ccccc3c2Cl)c1C c1(C(N(C)CC2(CNC(C3OCC4CCCC34)=O)CC2)=O)cc2ncccc2s1 c1(OC)ccc(CN2CCCCC2C(C)(C)O)cc1Cl c1(-c2nnc(CC(C(=O)NC3CCCCC3)N(C)C)o2)ccc2c(c1)OCO2 C1(NC(Cn2c(C)ccn2)=O)CCN(C(c2cccc(C(F)F)c2)=O)C1C C12(CNC(c3cc(SC)oc3)=O)CC1CN(C(=O)CCC1CCCO1)C2 C1(NC(=O)CC(C)C)CCN(CCN)CC1.C1(CC)CCCN1CC C1(CC(=O)NC2CC(CNC(C3CCCN(C)C3)=O)C2)SC2=NCCN2C1=O Cc1nc(C2CC2)[nH]c1C(=O)N(C(CNC(=O)Cc1cccnc1Cl)C1CC1)C N1(C(C(CN(C)C)(F)F)=O)CCOCC(C)(CNC(C2CCCSC2)=O)C1 c1(SCC(C)Cc2ccccc2)ccc(Nc2cccnc2)nc1 n1(CC(=O)N(C2CCN(C(=O)CCCn3ccnc3C)C2)CC)nnc(=O)[nH]1 N1(C(CC(C)N(C)C)=O)CCCC(C)(C)C1CNC(C1(C2CCCCO2)CC1)=O c1(N(C(=O)C(N)CCOCC(F)(F)F)C)ccc(C#N)cn1 c1(OC)cc(F)c2c(C(=O)N(CC(C)NC(=O)Cc3ccsc3C)C)n[nH]c2c1 C(=O)(CCC1=NNC(=O)CC1)NCC(=C)CCNC(=O)CCc1cccs1 C(CCSC)(C(=O)NCC(c1cccc(Cl)c1)NC(c1cc(F)n[nH]1)=O)OC n1(CCC)ncc(C(=O)N(C)CC2CCCCN2C(=O)C(C)C2CC2)c1Cl c1(N2CCC(CNC(C(C)O)=O)C23CC3)ncc2c(n1)COC2 c1(NCc2cc(C)c(Cl)nc2)[nH]c(=NCC(C)Sc2ccccc2)nc2sccc12 c1(C(=O)NCC(CNC(CCCC#CC)=O)F)cc(C)c(C)cc1Cl N1(C(=O)CCCc2cc[nH]n2)CC2(CCN2C(c2ncccc2Cl)=O)C1 C1(C(C)C)CC(O)CN1C(=O)CC1CCC(NC(C2COCC2(C)C)=O)CC1 N1(C(CCOCC)=O)CCC(O)C1C(N1CCOC(C2CC2)C1)=O C(C1CSc2ccccc21)N1CCN(c2ncnc(-c3ccccc3)c2)CC1 C1(CNC(C(N2CCCCCC2)C)=O)CN(C(=O)C(F)CC2CCC2)CCCO1 c1(C(=O)NC(C2CCCC2)CNC(C2N(S(C)(=O)=O)CC2)=O)c(Cl)n[nH]c1C1CC1 C(N=c1nc2c(ncn2C(C)C)c(N2CCC(C3CC3)C2)[nH]1)c1cnc(C)n1C N1(C(C(=O)NCC(C)SC)=O)CCOCCC1c1ccccc1 C1(C(N2CC(CC)NC(=O)C2)=O)N(C(=O)C=CC(F)F)CCCC1(C)C C1(C(=O)NCCCNC(C(C)OCCCCCC)=O)CC(=O)N(C(C)C2CC2)C1 C1(CNC(C(CN(C)C)(C)C)=O)CN(C(c2nnsc2N)=O)CC12CC2 C(Cc1ccoc1)(C(=O)NCC#CC1CC1)NC(=O)Cc1csnn1 C(=O)(C(CO)C(F)(F)F)N1C(C)C2CC1C2NC(C1CCCN1C=O)=O CCC(CC(=O)NCC#CCNC(C1(C)CC1(F)F)=O)C(F)F N1(C(CN(CCC#C)C)=O)CC(CNC(c2cccc(F)c2)=O)C(C)C1 Cc1ccc(C(=O)NC2CC(NC(c3c[nH]nc3C(F)(F)F)=O)C(O)C2)cc1C CCC(C)C(O)C(=O)NC1CC(F)(CNC(C2(CC(F)F)CCC2)=O)C1 C1(NC(C2COCCO2)=O)CCC12CN(C(=O)Cc1cccc(C(F)F)c1)C2 c1(OC)ccc(C(O)C(=O)NCC(C)NC(=O)C(=O)N(C)C)cc1 c1(NCc2ncc(CC)s2)cc(N(C)CC2(OC)CCCC2)ncn1 N1(C(CC(OCC)OCC)=O)CC=CC1(C)C(=O)NCCC(C)(C)CC N1(CCCC(=O)NC(CC)CNC(C2CC2C(N)=O)=O)C(=O)CNC1=O C1(NC(=O)CC2C=CCC2)CC2CN(C(c3cc(F)cc(F)c3)=O)CC12 c1(C(N2C(C)CCC(CNC(C3C(C)CCCC3)=O)C2)=O)ccc2ccnn2c1 N1(C(COCCCCOC)=O)CCC(C(O)CNC(=O)C=CC(=O)N(C)C)CC1 C1(C(N2CCCC(C(=O)CNC(C)=O)C2)C(=O)NC(CC)C)CC2CC1C1CC21 C1(C(=O)OC(C)C)N(C(=O)CCCc2cccc(Br)c2)CC12CCC(F)(F)CC2 CC1CN(C(=O)CCCC(F)(F)F)CC(C)C1NC(c1occc1F)=O C1(CC(C)NC(CCC=CC)=O)CCN(C(c2ccccc2SCC#N)=O)CC1 c1(NC(N2CC(n3cc(CC(C(C)C)O)nn3)C2)=O)ccc(Cl)c(SC(F)F)c1 CC(=O)CCCC(C)C(=O)NC1CC(CNC(C23CCC(CC2F)C3)=O)C1 Cc1cc(CNC(=O)C(C)(C)C)oc1NC(=O)C(=O)NC(CO)CCC1CC1 Cc1cccc(CC(N2CCC(CNC(C3CN(C)C(=O)N3)=O)C2)=O)c1C C1(C(N2C(CN(C(=O)CCCc3cnn[nH]3)C)CCC2)=O)C2CCC(C2)C1(C)C c1(NC(N2CC(OC)C(C)C2)=O)cc(C(=O)OC)c2c(c1)COC2 N1(c2nccc(CC#N)n2)CCC2C(CCCN2C(=O)CCCCN(C)C)C1 C(C(CC(=O)NCC(C)(Cn1cccn1)NC(c1cnc(Cl)s1)=O)C(F)F)OC C1(C(CNC(c2cc(CC)[nH]n2)=O)F)CCN(C(=O)C(C)CC2CCC2)CC1 C1(CC)CCN(C(=O)OC(C)(C)C)C1C(=O)NCc1ncc(C(F)F)cn1 C=CCC(CC=N)C(=O)N1CCC12CN(C(=O)C(C#N)c1ccccc1OC)C2 CCC(CC(=O)N(C1CCN(C(=O)CSc2nnnn2C2CC2)CC1)C)SC CCC(O)C(=O)NCCC1CCC(NC(=O)C=Cc2ncco2)C1 C1(N(C)C(c2ccc(-c3ccco3)s2)=O)CCC(NC(C2COC2)=O)C1 c1(CC#C)cccc(C(N2CC(C)C2C(=O)NC(C#C)C(C)OC)=O)c1 C1(C(N(CCNC(C2(OCC)CCOCC2)=O)CC)=O)C2CCCCCCC12 c1(OC)ccc(-c2nc(C3CC34CC4)nn2Cc2cccnc2)cc1OC N1(c2c3ncn(C(C)(C)CO)c3ncn2)CC2CCCCCC2C1 c1(-c2nnc(C=Cc3cccc(C#N)c3)o2)cccnc1S(C)(=O)=O C1(C)(CNC(c2ccc(C)nc2C)=O)CN(C(=O)CC2CCC2(C)C)C(C)(C)C1 c1(C(=O)NC(C2(O)CCN(C(=O)CC3CC(=O)NC3=O)C2)C)cc2n(c1)CCC2 C(=O)(C(CNC(c1csc(C)c1)=O)C(C)(C)C)NCCSCCCC Cc1nc2c(s1)CN(C(=O)C(C1CCOC1)NC(=O)CN1CCCC1=O)C2 C(=O)(C(CC(C)C)NC(=O)C(C)CCN(C)C)NC(CSC)C c1(C(=O)NC2CCC(NC(CCOCCCOC)=O)C2)cc(C)c(C)cc1Cl C1(C)(NC(c2cnc(CC)o2)=O)CCCCC1C(=O)NCc1conc1C C1(C(=O)NCC2CCSC2)CCCCCCN1C(=O)Cc1ccsc1 C(=O)(C1(C)COc2ccccc21)NCC1CC(NC(CCC(C)OC)=O)C1 N1(C(c2c(F)ccc(C)c2Cl)=O)CC2(CCN(C(C34CCC(CC3)C4)=O)CC2)C1 C(=O)(CC(C(C)C)NC(C1CCC1(F)F)=O)N1CCC(=C)C1 N1(C(C(=O)NC(C(CC)C)=O)C2CC2)CCOCC1CCCCOC(C)(C)C C1(C(=O)OC)CCC(CC)N(C(=O)CCNC(=O)OC(C)(C)C)C1.c1nnnn1C C1(NC(C2C(CCOC)C2)=O)COCC1C(=O)N(CCCc1cnn(C)c1)CC C1(NC(CCC#C)=O)CN(C(c2nc3cnccc3s2)=O)C2(CCOCC2)C1 Cc1cccc2c(C(=O)NC(C)(CNC(C3CC(C)N(C)C3)=O)CO)csc12 c1(C(=O)OC(=O)NC(C(c2cncn2C)N(CC)CC)=O)c[nH]c2c(Cl)cccc12 C1(OC)CC2CC(C(N3CCCC3CCNC(=O)C(C(C)C)C3CCC3)=O)CC12 C1(NC(=O)CCN)(CF)CCN(C(=O)CO)C1.c1(COC)cncc(Br)c1 CC1CCCC=C1C(=O)NCc1ccsc1C(=O)NCC1CC(=C2CC2)C1 c1(C(N2CC(CNC(C(COC)(C)OC)=O)OCC2)=O)cc2sc(C)cc2[nH]1 N1(C(CCSCC)=O)CCN(C(=O)C(C)(C)N2CCOCC2)CCC1C.CC(C)CCO C1(F)(CNC(c2cccnc2-n2ccnn2)=O)CCCN(C(c2cnsc2)=O)C1 O=C1NC(Cc2cccc(Br)c2)C(=O)N1CCCC1CC=CCC1 C(=O)(CC(F)(F)Cl)NCCN(CCC)C(c1csc(COC)n1)=O c1(NC(CNC2C(CS(C)(=O)=O)CC2)=O)nc2c(F)cccc2o1 N1(C(CC(C)N(C)C)=O)CCC(NC(=O)C(c2cncnc2)C)C(O)C1 c1(C(N2C(CNC(C3C(CC)CCO3)=O)CC(F)C2)=O)cc2cccnn2c1 S(=O)(=O)(c1cccc(-c2nn[nH]n2)c1)NC(CC(c1cccc(OC)c1)SC)=O CCCC(C(F)(F)F)NC(=O)CC1CCC(NC(=O)CCCCOC)CC1 N1(C(CNC(CC(C)C)=O)=O)CCOCC(C(=O)NCC(C)(O)C(C)C)C1 C1(=O)C(F)(F)CC(OC)C(=O)N(C)CC(C)N1.C1(C)CCCOC1.OC N1(C(C2CC(C)OCC2)=O)CCN(C(C2(Cl)CC2)=O)CC2(CC2)C1 CC1OC(=O)NC1C(=O)NCCCCCNC(c1ccn(CCN(C)C)n1)=O N1(C(c2c(CCC)n[nH]c2)=O)CCOC2(CCCN(C(=O)C(F)=C3CCC3)C2)C1 c1(CCCC)ccc(C(=O)NC2COC(C(C)C)C2)c(C)n1 C#CCCCCCCC(=O)N1CCCC1(C)C(N1CCOC(C(C)C)C1)=O C1(CC(c2ccc(C(C)(CO)OC)o2)OC)CC(C)(C)NC1=O C(C(CNC(=O)CCSc1ccccn1)S(C)(=O)=O)NC(c1c(CC)nn[nH]1)=O c1(CC)ccc(Cl)c(C(N2CCOCC(NC(C3CCS(=O)(=O)N3)=O)C2)=O)c1 C1(NC(COC)=O)CCCN(c2nnc(C(C)(C)O)n2CC2=CCCOC2)C1 N1(C(c2c(C)nns2)=O)CCC(C(=O)NCCN2CCC(CO)C2)(C(C)C)C1 c1(CC(=O)N(C2CCC(NC(c3cccnc3)=O)C2)C)ccn(CC(F)(F)F)n1 C1(C(=O)Nc2cccnc2Cl)COCCN(C(=O)C(F)(F)CO)C1 c1(CC(=O)NCCCN(C(C)C)C(c2c(C#N)cnn2C)=O)ccc(F)c(F)c1 C(=O)(C(C)(C)CC(=O)NCC(C(=O)NCCCCCC1CC1)C(C)C)OC C(=O)(C(C)P(C)(C)=O)NCCCN(C(C(c1ccc(C)o1)C)=O)CC1CCCC1 CON(CCC(=O)N1CCn2c(C)nnc2C1)C(=O)C1CCCCC(=O)C1 c1(OC(C)C(=O)NC2CCN(C(=O)CCC3CC3)C2C)ccccc1Cl c1(C(=O)NCC2CN(C(C3CC3C3CCC3)=O)C2)ccc2cnccc2n1 N1(C(c2csnn2)=O)CCCN(C(c2cnc(-c3ccccc3)s2)=O)C(CO)C1 CCC(CC(C)C)C(=O)N1CC=CC1CNC(=O)Cc1cccc(Cl)c1F C1(CN2C(c3cc(C(=O)OC)no3)CCCC2)CCCC2(CCC2)O1 n1(CC(=O)N(CCNC(C(C(C)C)F)=O)C)cnc([N+](=O)[O-])n1 c1(C(N2CCC(N(C(c3c(C)cnnc3)=O)C)C2)=O)cc(N)nc(Br)c1 c1(C(=O)Nc2nccc(C(N3CCN(C)CC3)=O)c2)cccc(C#CCO)c1 N(C(=NCCC(=O)N(C)C)NC(c1c(F)cccc1F)C)CC1C(C)C1 C(=O)(C1=CS(=O)CCC1)NCC12C(CN(C(CNC(CNC(C)=O)=O)=O)C1)CC2 c1(C(=O)NC(CC=C)CNC(c2ccc(=O)n(C)n2)=O)ccc(N=S(C)(C)=O)s1 N1(C(CC2(CSC)CC2)=O)CCC(NC(=O)Cc2cocn2)CC1C1CC1 C(=O)(C(CC(=C)C)NC(C1CC1C(F)F)=O)NC(C1CCOC1)C#C CC1CCOC1CC(=O)NCC(C)(C)O.C(C(=O)N(CCCN(C)C)C)OC1CCC1 CCC(F)C(=O)N1CC(C(C)NC(=O)C(N2CCCCC2)C)C1 N1(C(C(C(CC)C)O)=O)CCC2(CCC2)C(NC(c2cc3c[nH]cnc-3n2)=O)C1 C1(NC(C2=CC(C)(C)C2)=O)CC12CCN(C(C1CC=CC1)=O)CC2 C1(C(N2C(C)(CNC(c3c(OC)nccc3)=O)CCC2)=O)CCCC12OCCO2 c1(CCn2cc(C3CCN(C(C)=O)CC3)nn2)ccc2c(c1)CC(C)O2 C1(CN(C)C(C2CCC(F)(F)C2)=O)CN(C(=O)OC(C)(C)C)CCO1 N1(C(=O)Cc2ccsc2)CCC(C2CCN(C(C34CC3C4)=O)CC2)C1 C#CCCCCCCCNC(=O)C(CCC1CCC1)NC(=O)C(C)C c1(C(N2CC3C(NC(C(C)N(C(C)=O)C)=O)(C3)C2)=O)cc(C#N)c(F)cc1F c1(OC)ncccc1C(=O)NC(CNC(=O)C(C)Oc1ccc(F)cc1)C(C)C C1(OC)CC(CNC(=O)Cc2scnc2C)N(C(=O)CCSC)C1 C1(NC(C2(OC)CCC2)=O)CN(C(C2CC3CCC2C3)=O)C2(CCOCC2)C1 C1(C(=O)NCC(C)(O)C(F)F)(NC(CN(C)C)=O)CCc2cc(Br)ccc2C1 N1(C(C(C)CS(C)(=O)=O)=O)CCC2CCCC(C1)N2C(c1csc2nnsc12)=O Cc1nn(C2CC2)cc1C(=O)NC1(C)CCN(C(c2coc(Cl)n2)=O)C1 C1(NC(Cc2cc(C)sc2C)=O)CCN(C(=O)C=Cc2cnc(C)s2)C(C)C1 C1(CC=C)(C(=O)NCCSCCO)CN(C(=O)C=CC(N2CCOCC2)=O)C1 c1(C(=O)NCC(C2CCC2)NC(COC(C)C)=O)cnoc1-c1cccs1 C12CCCCN1C(=O)CSCCC(=O)NCC2.S(C)(=O)(=O)NCCC c1(C(N2CC(F)(CNC(C(C)OCC)=O)C2)=O)cc(C2CC2)nnc1O N1(C(C(OC)OC)=O)CC(CNC(=O)C2=COCC2)C(c2ccccc2)C1 c1(C(=O)NC(CC2CN(C(C(C)CSC(F)(F)F)=O)C2)C)cc2ccsc2[nH]1 CC1CN(C(=O)C=CC2CCN(C(=O)CC3COCCO3)CC2)CC(=O)N1C CCC(CC(=O)N1CCC(C)(CNC(C2CC(=O)OC2(C)C)=O)C1)C(C)C c1(CC)ncc(C(=O)N(C(C)C(=O)N(CCCC(=C)C)C2CC2)C)cn1 n1(CC(=O)NC(CN(C(C2CCCC23CC3)=O)CC)C)c(=O)oc2ccccc12 N1(CC(N2CCC(Cc3cn(Cc4cn(C)nc4)nn3)C2)=O)C(=O)COCC1=O c1(C(N2CCC3CN(C(=O)C(F)(F)C4CC4)CC23)=O)cncc2cc(Cl)ccc12 C(CSCNC(C1(Cl)CC1NC(C)(C)C)=O)(C(=O)OC1CCCCC1)OC(C)=O CCC(CO)C(=O)NCC1CN(C(=O)CC2COC(C)(C)C2)CCO1 c1(C(N2C(CCNC(C3C(=C)C3)=O)CC(F)(F)C2)=O)cc2cc(Cl)ncc2[nH]1 C(=O)(C(C)CC(F)F)N1CC(C2CN(C(C3(SC)CCC3)=O)C2)OCC1 N1(CCCNC(CC2N(C(CCN(C3CCC3)C)=O)CCC2)=O)CCS(=O)CC1 N1(C(CC(C(C(C)C)C)C)=O)CCC2CC(CNC(=O)C3=CCSC3)CCC2C1 N1(CC(=O)N(c2ccnc3ccccc23)CCO)CCN2CCCC2C12CCC2 C#CCCC(O)C(=O)NCc1nc(CNC(c2cc3occc3[nH]2)=O)cc(O)n1 N1(C(COCCCC)=O)CCN(C(=O)Cc2cc[nH]c2)C(C)C1 C1(NC(C2(C)CN(C(C(C)N(C)C)=O)C2)=O)CCC(C2CC2)C1 Cc1cc(=O)c(C(N2CCC2c2cn(CC3CCC(=O)O3)nn2)=O)c(C)[nH]1 c1(-c2c(COC)cncc2)cccc(N=S2(=O)CCCC2)c1 N1(C(CC2CC(OC)C2)=O)CCC1C=CC(C)(C)C.C1C(=O)N1C C(=O)(CCCCC(C)(C)C)N1C2(NC(COC)(C)CC(=O)O)CC(C1)C2 CC1CCOCC1C(=O)NCCCCNC(=O)CN1CCC(CO)CC1 c1(C(=O)NC(CC(C)C)CNC(=O)CC2CC(F)C2)cccc2cc(O)ncc12 C1(NC(C(c2ccccc2)NC(C)=O)=O)CN(Cc2ccc(C)cn2)CC1O c1(OCC)ccc(CCCC(=O)NC2CC2NC(=O)CCSC2CC2)cc1.C1(O)=CN=C1 C1(C(=O)NCCCNC(c2n(C)nc(C3CCC3)c2)=O)CC12CCC1(CC1)CC2 c1(CC)ccc(C(=O)NCC2(O)CN(C(C3CC4C=CC3C4)=O)C2)c(Cl)c1 C(CC(C)C)(C(=O)NCC1(O)CC(C(=O)NCC2CC(C(C)(C)C)C2)C1)OC C12(C(=O)NCC(C)NC(C3ON=C(C)C3)=O)CCCC1CCC2 c1(C(=O)NC2CCN(C(c3c(C)cc(C)c(C)c3)=O)C2)cc(S(N)(=O)=O)c(C)o1 N#Cc1cc(C(=O)NC2(CCC(=O)NC3CCNC(=O)C3)CCCC2)c[nH]1 c1(C(=O)OC)cc(NC(=O)CCc2ccon2)cc(OC)c1C N1(C(c2c(N)ccc(Cl)c2)=O)CCC2(CNC(c3cc[nH]n3)=O)CCCCC12 CCC(C(=O)N(C1CN(C(=O)COc2ccc(OC)cc2)C1)C)C(C)(F)F c1(C(C(=O)NCCN(C(=O)Cc2cc(C3CC3)no2)CCC)C)ccccc1F c1(C(=O)NCC(C2CCN(C(C(C)SC)=O)CC2)C)cccc2nccnc12 c1(C(N(C2CCN(C(=O)CC3OCCO3)C2)CC)=O)c(F)cccc1F c1(CC)cc(OC)ccc1C(N1CCC(CN(C(=O)C(C)(C)C#N)C)C1)=O n1(C(N2CCC2CF)=O)cc(C2CC2COC2CCOC2)nn1 N1(C(C(COC)O)=O)CC2(c3cn(CCCOCC(C)C)nn3)CC1CCO2 C(CCNC(=O)C(C1CCCCCC1)C)(C(C)(C)C)NC(c1c(C)cncc1)=O C(CCC(O)C(=O)N1CCOC(C#N)C1)NC(c1nc(C)oc1C)=O C1(NC(C(C)(C)NC(=O)CC2CC(=O)C2)=O)CCC(=O)NC1(C)C C1(NC(CCC(=C)Cl)=O)CN(C(c2ccccc2C(F)(F)F)=O)CC(C)(C)C1 C12(NC(CCCC#C)=O)CC(CO)(C1)OC21CN(C(C2(CC3CC3)CC2)=O)C1 CCC(CN(C)C)CC(=O)N1CCC1C(=O)NCC(=O)NC C1(C(C(=O)NCC=CCNC(C2(CC3CC3)CC2)=O)O)CCS(=O)(=O)CC1 C(CN=c1[nH]c2cc(Cl)ccc2s1)NC(C=C1N(C)C(=O)CS1)=O N1(C(C(CCC)C(=O)O)=O)CCOC2(CCN(C(=O)C(F)(F)F)CC2)C1 Cc1cccnc1C(N1CCCCC1CCCNC(c1nocc1C1CC1)=O)=O C1(NC(c2cncc(NC)c2)=O)CN(C(=O)CC2CCCC(=O)N2)CC12CCC2 c1(C(C(=O)NCC(CNC(C(C(=C)Cl)(C)C)=O)(C)O)(F)F)nc2ccccc2s1 c1(C(N2CC3CC(NC(C4(CCO)CC4)=O)CC3C2)=O)noc2c(F)cccc12 C1(NC(CC=CC)=O)CC2CC(C1)N(C(=O)COc1ccc(C(=O)NC)cc1)C2 c1(-n2c(CC3CCC(=O)NC3)nc(-c3ccccn3)n2)ccc(F)cc1F CC1CCN(C(=O)CN2CCN(C)CC2)C(C(=O)NCCN2C(=O)CNC2=O)C1 C1(C(C)C(=O)NCCn2cncn2)CCN(C(=O)C(C)(C)CC2CC2)CC1 c1(C(=O)NCCOCCN(C(C2CCC(C)O2)=O)C)cccc(C(=O)C2CC2)c1 CC(CC(C)(C)C)C(=O)NC1CN(C(c2cnc3ccccn23)=O)CC1C(F)F c1(N2C3CC(CC)CC2CC3)ncnc2n[nH]c(C)c12 CCC(CNC(C1(COC)CC1)=O)N=c1[nH]c2ccc(Cl)cc2s1 N1(C(COCCC(C)C)=O)CCC2CN(C(=O)Cc3ccc(Cl)c(Cl)c3)CC2C1 CCCCCCCCNC(=O)NC(C1CCCC1)CS.C1(Br)(CCO)CC1 C(CCC)(C(O)C(=O)NCc1cccnc1C)NC(C(C)OCCC=C)=O Cc1ccccc1C(C(=O)O)NC(=O)C=CC(=O)N(c1nccs1)C C1(N(C(C(C)=CC)=O)C)CN(C(c2nn(C)cc2N)=O)CCC1O c1(C(N2CCC(O)(C(C)CNC(C34CCC3CC4)=O)C2)=O)c[nH]c2cnccc12 c1(C(N(C(CCNC(C(C)NC(COC)=O)=O)C)C)=O)cc2cc(F)ccc2o1 c1(SC)ccc(C(N2CCCC(CCNC(C3(CF)COC3)=O)C2)=O)cc1 Cc1cc([N+](=O)[O-])cc(C(=O)NC2C=CCN(C(C3(O)CCOCC3)=O)C2)n1 C(CC(C)C(=O)NC(CCN(C)C(C1(C(C)C)CCC1)=O)C(C)C)=CCC c1(C(N(C2CCCN(C(c3ccsc3)=O)C2)C)=O)ccc(Cl)c(O)c1 C12C3CC4C(C3NC(=O)C(=O)N3CC(C3)COC1=O)C24.c1(OC)ccccc1.CO c1(C(N(CC(CN(C)CC2CCC(F)(F)C2)O)C)=O)cc2n(n1)CCO2 C1(C(=O)N(CC(C)NC(=O)CCc2ccnc(C)n2)C)(OC)CCC(C)(C)C1 C1(CCC)CC(NCCc2cccc(F)c2)CCO1 C(=O)(CCCCCCCC1CC1)NC(CCCNC(C1=C(C)OCC1)=O)C c1(C(N2C3CCC(NC(c4ccc(C=C)cc4)=O)(C3)C2)=O)cc2cc(Cl)sc2[nH]1 C1(NC(c2n(CCN(C)C)ncc2)=O)CN(C(c2cc[nH]c2)=O)CCC12CCC2 c1(SC)ncc(CCC(N2CCC(CNC(C3CN(C)CCO3)=O)C2)=O)c(O)n1 c1(OC)cc(CNC(=O)C(N2CCCC3(CC3)C2)c2ccc(F)cc2)ccc1OC c1(OC)cccc(CC(C(C)C)NC(=O)NC2CSC(C)(C)C2)c1 c1(CN(C(CCC)C)Cc2ccccc2)ccc2c(c1)CCCN2C C1(C(=O)NC2CCN(C(c3c(C)cc(C)[nH]3)=O)CC2C)CCc2nccn2C1 N1(C(C(c2cccnc2)NC(C)=O)=O)CCOC(CNC(=O)CC2C=CCC2)C1 c1(OC)cc(C(O)C(=O)N2CC(NC(=O)CC(C)F)C2)c(F)cc1O c1(NC)nc(C(N2CCC(NC(=O)C3CC3)C2(C)C)=O)ccc1[N+](=O)[O-] C(CC(=O)O)(CC(C)C)NC(c1c(Nc2nc(C)sc2)cccc1)=O C(CCCCCNC(=O)CN1CCCCC1=O)NC(C(CC)c1cccnc1)=O N1(Cc2cn(CCC(C(C)C)NC(=O)CCC(F)(F)F)nn2)CCc2ccccc21 c1(C(C)NC(C2(n3cc(-c4scc(NC)n4)nn3)CC2)=O)nc2c(s1)CCCC2 c1(CN2CCCC(C(N(C(C)C)C)=O)C2)cccc2ccnn12 c1(CC(N2CC(F)(CNC(CC3C(CC)C3)=O)C2)=O)c[nH]c2c(F)cccc12 C1(CCNC(C2(CC)CC2(F)F)=O)CCCN(C(=O)CCc2ccsc2)C1 CC(CC(F)(F)F)C(=O)NCCCN(C(=O)Cc1nc[nH]n1)C1CC1 C1(NC(c2c(C)sc(Br)c2)=O)CC(C)CN(C(c2nonc2N)=O)C1 C#CCCCC(=O)NC1CC(CO)N(C(C2CCOC(C)(C)C2)=O)C1 c1(C(=O)NC2CN(C(Cc3ccc(C)cc3)=O)CC2C#N)cccc2ccnn12 C1(C(F)(F)F)(NC(=O)NCCC2(c3ccccc3)CCOC2)CCOC1.C(CO)S C1(C(=O)OC)C(C(=O)OCC(=O)Nc2cccc(F)c2)C2CCCCCC12 c1(C(C(N2CC(N(C)C(C3CC3F)=O)C2)=O)O)cccc([N+](=O)[O-])c1 N1(C(C(C(C)C)N(CC)CC)=O)CC2CCCC(C1)N2C(=O)C(C#N)C1CC1 C1(CC(N2CC(C(N)=O)(OC)C2)=O)CCN(C(=O)Cc2cc[nH]c2)C1(C)C C(=O)(C(C(C)C)c1ccc(Cl)cc1)N(CCN(C(CNC(=O)NC)=O)C)C1CC1 Cc1cccc(C(N2CCN(C(C3CC3C3CC3C)=O)C(C)C2)=O)c1C(F)(F)F c1(OC)ccc(Cl)c(C(N2CC(F)(F)CC2CNC(C2CCCS2)=O)=O)n1 CCC(C)C(C)C(=O)NC1CC(F)(CNC(=O)COc2cc(F)cc(Cl)c2)C1 C1(NC(=O)CCc2cnc[nH]2)CCC2(CCN(C(=O)C(C3CCCCC3)F)C2)C1 n1(C(CC)C)ccc(=NC(=O)CCNCCCC2CCC(F)C2)[nH]1 c1(C(=O)NCC2CCN2C(c2coc(CO)c2)=O)ccc2c(n1)CCC2 c1(CC(C(=O)NCC(C)NC(C2(CC)CC(C)(C)C2)=O)C#N)ccc(C#N)cc1 C12(NC(CCc3n(C)ccn3)=O)CC(C1)N(C(=O)Cc1ccsn1)C2 C(=O)(C(CC(C)C)ONC(=O)C=CC1CCC1)NC(C(=O)OC)C c1(CC)cc(F)c(C(N2CCCC2CNC(=O)C(C)C(=O)OC)=O)cc1F C1(NC(C2N(C)C(=O)OC2)=O)CCCCN(C(=O)CNC(=O)CCC2CCCC2)C1 CC1CCN(CCO)CC1NCc1ccccc1.c12sc-1nc2C(F)(F)F N1(Cc2nc(C)c(Br)s2)CC2(CNC(C3CCCC3O)=O)CC1CO2 N1(C(c2c(CC)nc(C)[nH]2)=O)CCC(CNC(C2(C#N)CCCOC2)=O)C(C)C1 c1(CNC(C23CC(NC(c4c(C)n[nH]c4)=O)(C2)C3)=O)cc2ccoc2cn1 C(=O)(C(O)C(C)(C)C)N1CCC(O)(C(C)NC(C(C)C(F)F)=O)C1 c1(C(N2CCC3CN(C(C(C)OC)=O)CC32)=O)cccc([N+](=O)[O-])c1F c1(C(=O)NC2CC(C(N(C)CC3(O)CCC3)=O)C2)cnn2ccccc12 Cn1cc2ccc(CN3CCC(C(=O)Nc4ccc(C#N)nc4)C(O)C3)cc2n1 Cc1cccc(O)c1C(=O)NC(C)CCCCNC(C1CC(=O)N(C)C1)=O c1(C(=O)NC2CCC(NC(c3n[nH]cc3Cl)=O)CC2)cc2n(n1)CCCCC2=O N1(C(c2cn(CC)nc2)=O)CCC(C)(C)C1C(=O)NC(CO)C1(C)CC1 CC1(C)COCC(C(N2CCN(C3CN(C(C4(C(N)=O)CCC4)=O)C3)CC2)=O)O1 C1(C(c2noc(C3(C4CCCCO4)CCOCC3)n2)C)CCN(CCO)CC1 CC(C(=O)N(C1CCN(C(C)(C)C)CC1)CCO)C1=CCCC1.C12CC(C1)OC2=O C1(NC(=O)Nc2cc(C)nn2CC2CC2)CC1C1CCCC1 c1(CNCC(F)CC2CNC2)ccc(Cl)c(C(F)(F)F)c1 C(=O)(CCCC(C)(C)C(=O)OC)NC(c1ccc(CC)cc1)CNC(CC=C)=O S1(=O)(=O)c2cnc(s2)N1.c1(C(C(=O)OC)N(C)C(C)=O)ccccc1Br N1(C(CCCn2cc(CCN(C)C)nn2)=O)CCC(C2CCC(=O)N2)CC1 N1(C(C2(N(C)C)CCC2)=O)CCC(N(C)C)C1.C1(=O)C=CCN1 CCCCCCC(=O)NC1CN(C(=O)CCCN(C)C2CC2)CC1OCC N1(C(c2cccc(C(C)C)c2)=O)CC2(C1)CN(C(=O)C1=CCOC1)CC2CO c1(NC(CNC(c2c(C)cc(CC)o2)=O)C2CC2)cnc(C#N)cn1 c1(C(N(CC)Cc2cc(C)cc(C)c2)=O)cc2nnn(C)c2s1 c1(C(=O)NC2(C)CCN(C(C(CCCC)=O)=O)C2)cnn2cc(OC)ccc12 N1(C(Cn2ccc(C(=O)OC)n2)=O)CC2(CCN(C(C3(C)CCOC3)=O)C2)C1 N1(CC)CCCCC1C(N1CCCC1C(N1CCC(OC)C1)=O)=O S(=O)(=O)(c1cc(C)sc1[N+](=O)[O-])N1CC(C(=O)OC)CC12CCCC2 C#CCCCC(c1nnnn1CCCOC)NC(C1CCOCC1)C Cc1cc2[nH]c(C(=O)NC(CNC(c3coc(CO)c3)=O)C(C)(C)C)cc2o1 C1(C(=O)NC2CC(O)(CNC(CN(CCOC)C)=O)C2)Cc2ccc(F)cc2C1 c1(C(=O)NCC2C(CNC(c3c(C(C)C)ocn3)=O)C2)cc(F)cc(Cl)c1 CC1(C)CCN(C(=O)C(c2cccnc2)C2CCCC2)c2ccccc21 C(=O)(C(C)C(F)(F)F)N1CCC(CC=C)(C(N2CC(C)(CF)C2)=O)C1 C1(CN(C(=O)CSCCNC(c2sccc2Cl)=O)C)CCCC1O CC(C)CC(F)C(=O)NCC(C(C)C)NC(c1[nH]nnc1C1CC1)=O C(CCCC(=O)N1CCC(C(C)(C)CNC(C2CCOC(C)C2)=O)CC1)OC N1(C(C(CC)NC(C)=O)=O)CCC2C(CCN2CC2CCCN(C)C2)C1 C(C(CC(=O)N1CCCCC1CN(C)C)OC)NC(CNC(CC)(C)C)=O c1(C(=O)NCC2CN(C(=O)C=CCO)CCCO2)ccc2occc2c1 N1(C(C(N2CC3CC3(c3cccc(F)c3)C2)=O)=O)CCOC(c2ccccc2)C1 C1(CC(=O)NCC(C)CCO)CC2(CC2)CN1C(=O)CC1(O)CCCCC1 C(=O)(CCC(F)(F)C(F)F)N1CCN(C(C(C)C2CC2)=O)CC(O)C1 CC1CCN(C(=O)C=C(Cl)Cl)C(C)C1NC(c1cc(O)no1)=O c1(OCC(=O)NCC(CC)NC(C2CC2c2cncn2C)=O)ccncc1 C1(COC)(NC(c2cnc(CC(C)(C)C)s2)=O)CN(C(C2CCC(C)S2)=O)C1 N1(C(c2ccc(N)c(O)c2)=O)CC(NC(=O)CC(=O)NCC(F)F)CCC(O)C1 C1(C(=O)NCC(CN(C(=O)C(c2ccccn2)O)C)(C)C)CC(=O)C1(C)C CC(C)CC(F)(F)C(=O)N1CCC2(CC1)CC2CNC(=O)C#CC1CC1 CC1CC(C(=O)NCC=C2CCN(C(c3ccccc3Cl)=O)CC2)C(=O)O1 Cc1cc2[nH]c(C(N3CC(C)C(C)(C(N4CCOCC4CO)=O)C3)=O)cc2o1 S(=O)(=O)(c1ccc(C)cc1Cl)NCC.C1(=O)CS(=O)(=O)NC2C(C2)CO1 N1(C(c2cnc(CC(C)C)s2)C(=O)NC(C)C)CCn2ncc(S(C)(=O)=O)c2C1 c1(NCC2(CNC(C(CC)(C)OC)=O)CC23CCC3)ncnc2sc(C)nc12 c1(C(=O)NC2(CN(C(c3c(C)nccc3)=O)C)CC2)cc2c(F)ccc(F)c2[nH]1 c1(C(N(CCCCN(C(c2cc(OC)no2)=O)C)C)=O)ncncc1C c1(C(=O)NC2CCC(F)(CNC(CCC(C)OC)=O)C2)[nH]c(C)c([N+](=O)[O-])c1C c1(C(N(C)CC2(O)CN(C(C(C)CCN(C)C)=O)C2)=O)cnccc1C#N Cc1ccccc1CC(N1CCC(C)(NC(c2cn(C3CCOC3)cn2)=O)C1)=O CC1CN(C(C2CN(C(c3cnccn3)=O)CC2(C)C)=O)C(C)C1C c1(C(N2CC(COC)(NC(=O)CSS(C)(=O)=O)C2)=O)c(C)cc(C)cc1C CC(c1ccc(F)cc1)=CC(N1CCN(CCCNC(=O)C#CC2CC2)CC1)=O c1(C(=O)NCC2C(NC(c3ncn(C)n3)=O)C2)cnc2c(N)cccc2c1 c1(C(N2CCC(c3nncs3)C2)C(=O)NCCSC)nc(C)c(Br)s1 CC1CN(C(=O)Cc2csc(C3CC3)n2)CCCN1C(C1COC2(CCC2)C1)=O Cc1cnc2cccc(C(=O)NC3CC(C)CN(C(c4ncsc4C)=O)C3)n12 C(CNC(=O)Cn1cnc(C(F)(F)F)n1)(C(C)C(C)C)NC(CCNC(C)=O)=O C(=O)(C(C)CC(F)(F)F)NCC1(OC)CCN(C(C(C=C)(F)F)=O)C1 c1(C(N2CCCCCC2CNC(C2(O)CCSCC2)=O)=O)cn2cnnc2cn1 C1(C(N(C2CCC2)CC=CC(C)(C)C)=O)CN(C(C2CCC2)=O)CC(C)(C)C1 N1(C(C(C(CC)CC)C)=O)CCC2(CCN(C(c3ccccc3C(C)C)=O)C2)C1 n1(CC(=O)NCCC2(O)CCN(C(CC3C(C)C3)=O)CC2)cc2ncccc2n1 Cc1ccc(CN2CCCC2SCC(=O)NCc2ncccc2C)c([N+](=O)[O-])c1 c1(C(N2C(C)CC(NC(c3c(CC)nco3)=O)C2)=O)cc(N)ccc1O Cc1c(CCC(N2CCOCC(NC(c3cnc[nH]3)=O)C2)=O)cccc1Br c1(N2CCC(OCC)C(C)C2)[nH]c(=NCC#Cc2cccnc2)nc2sccc12 c1(CC)cccc(CNC(=O)NCC(c2ccc(Br)c(F)c2)(C)O)c1F c1(OC)cc(N)c(Cl)cc1C(=O)NCC1CCN(C(C2CNC(=O)N2)=O)C1(C)C c1(C(=O)NCC2(COC)CN(C(C3CCCOCC3)=O)C2)ccc2nn[nH]c2c1 N1(C(C(c2cccs2)SC)=O)CCC(CNc2sccc2C(=O)NC)C1 c1(C(=O)NCCN(C(=O)C(O)CC(C)C)CC)ccc2c(c1)S(=O)(=O)NC2 N1(C(CCSC)=O)CC(NC(c2c[nH]nc2C)=O)CC(F)C1 C1(C(C)NC(C=CCOC)=O)CCCN(C(=O)CN2CCC(C)(C)C2)C1 c1(NC(=O)NC(C(=O)OCC)C)nn2ccccc2c1C(=O)NCCCCO CC1C(NC(=O)Cc2cccnc2)CCCN1C(c1cnc(O)nc1O)=O N(C(=NCCC)N1CCC(NC(c2ccccc2C)=O)CC1)C(C#C)CC c1(C(=O)NC2CN(C(c3cc(SC)c(C)o3)=O)CC2CO)c(C)nn(C)c1N Cc1sc2ccccc2c1C(=O)NC1CN(C(=O)C(C)(C)CO)CC1C c1(CC)ccc(C)cc1C(=O)NCC(O)CCNC(c1cc(N)cc(F)c1)=O N1(C(=O)NCCCn2c(C)ncc2)CC2CCC(C1)C(=O)O2 Cc1nccn1CCC(=O)NC1C(C(=O)NCCCC2CCCCO2)C1(C)C c1(N(C2CCCN(C(C3C(=C)CC3)=O)C2)CC(C)C)ccc([N+](=O)[O-])cc1 C1(C(F)(F)F)(C(=O)NCC(CC)NC(c2cc(C3CCC3)[nH]n2)=O)CCN(C)C1 c1(NC)ccc(F)cc1C(N1CCCCC1CNC(=O)CNC(=O)C(C)(C)C)=O c1(-c2cccc(OC)n2)cccc2cc(C(=O)NC(C3CCOCC3)C)sc12 C(=O)(C1CCCn2ccnc21)N1CCCC(C)(NC(c2csc(C(N)=O)n2)=O)C1 n1(CC#C)cccc1C(N1CCC1CC(=O)NC(CC)C(=O)OCC)=O C1(C(=O)NCC2CN(C(C3(CC#N)COC3)=O)C2)CC(=O)N(O)C1 C12CCCN(C1)CNC(=O)CC2.Cc1ncsc1CCNC(=O)OC(C)(C)C C1(NC(C2(N(C)C)CCC2)=O)CCCCN(C(=O)C(c2ccc(N)cc2)(C)C)C1 N1(C(CCCN(C(=O)OC)C)=O)CCOC2CN(C(=O)C(O)CC(C)(C)C)CC12 N1(C(c2cn(C)nc2)C(=O)NCC2CCCO2)CCN(C(=O)N(C)C)CC1(C)C Brc1c(-n2cnnc2)n[nH]c1-c1ccc(Br)s1.c1(C(CCl)N)ccccc1 c1(C(=O)NCCC2CCN(C(=O)CCCF)C2)cc(Br)n2ccccc12 N1(C(C=CCNC(=O)CCn2cccn2)=O)CCC2CCCCC12 C=CCC(CC(=O)N1CCCN(CCO)CC1)NC(C1(C)CCCCC1C)=O c1(OC)ccc(S(=O)(=O)N2CC(O)C2)cc1-c1ccnc(N(C)C)c1 CC1CCC(CNC(=O)COCC2CC2)N(C(C23COCC(C2)C3)=O)C1 C(=O)(C(C)(C)C1CCCCC1)NCCCNC(C1C(C)C1)=O C(CC(C)(C)C)(C(=O)NCCC1COCCO1)NC(CSCCC(C)C)=O C1(F)(CNC(C=CCN(C)CC)=O)CCN(C(=O)CC(=O)N(C)C)CC1 C1(NC(C2(CCOC)CC2)=O)CCN(C(=O)CCC2CCC(C(N)=O)O2)CC1C c1(NC(N2CCC(NC(=O)CCCC3CC3)C2)=O)cccc(Cl)c1F C(=O)(CCC1CC(NC(C2CCN2C(C)(C)C)=O)C1)N(CCCO)CC c1(C(=O)NC2C3CCN(C(COCC=C)=O)C3C2)ccc(S(=O)(=O)NC)c(F)c1 c1(C(=O)NCC2=CCCN(C(C(C(CC)(C)C)O)=O)C2)nn(C)cc1S(N)(=O)=O C(N=c1[nH]c(=NCc2ccc3c[nH]nc3c2)[nH]c2ccsc12)C1C(C)CCCC1 N1(C(=O)OC(C)(C)C)CCC(C2CC2)(C(=O)OCCNC(=O)C2=CCCC2)C1 C1(NC(=O)CCc2cncs2)CN(C(c2conc2C2CCCC2)=O)CCC1F C(=O)(CCC(=O)NCCC1CC(NC(=O)C(C)(C)CNC(C)=O)C1)NC c1(OC(C)C)cccc(C(=O)NC(C2CCCN2C(=O)CC(F)F)C)c1 c1(OC)c(C)nc[nH]c1=NCC1CN(C(=O)C(C)(O)C2CCC2)CC12CCC2 c1(CCC(=O)NC(C2CCCN2C(=O)C2CC2)C(=O)OC)ccc(C#N)cc1Br N1(C(=O)NCCN(C)C)CC(=O)NCC2(CCC2)C1 c1(C(N2CCC(O)(C(C)NC(Cc3cc(C)[nH]n3)=O)C2)=O)cc(O)cc(N)c1Cl C(=O)(C(C)(C)CC(=O)NC(C)(CNC(C1(C(=O)OC)CC1C)=O)C(C)C)OCC c1(C(N2CC(CN(C(=O)CC34CCC(CC3)CC4)C)C2)=O)cc(O)c(O)c(O)c1 CC1C(C)N(C(=O)COc2cccc(C#N)c2)CCN1C(c1cnccn1)=O N1(C(c2c(C)cccc2)=O)CCC(C2CC2NC(c2cc(C#N)c[nH]2)=O)CC1 c1(CC(C)C)ccc(C#N)c(NC2CN(C(=O)CC3CC(O)C3(C)C)C2)n1 C=CCC(C(=O)N1CCC(O)(CNC(=O)C=CCCC=C(C)C)C1)C(C)C CC(C)C(C)CC(=O)N1CC(N(C)C(c2cc(N)cc(O)c2)=O)C2(CC2)C1 c1(OC)cc(SC)ccc1C(=O)NC1COCC1NC(=O)CC1CCCC1 C1(C(=O)NCc2cc(C)sc2)CC(O)C(O)CC1CNC(=O)C(CO)NC(N)=O O=C(CCC(F)(F)Cn1cc(CCCO)nn1)NC(c1nccs1)C1CC1 c1(C(C#N)N(c2snc(C)n2)C(=O)CC2CCCC(O)C2)ccc(F)cc1F C1(C(=O)NCc2cn(CC)nn2)CC(NC(c2cc[nH]c2C)=O)C1(C)C c1(NC(=O)NC2C(C(=O)NCC(c3ccc(C)s3)C)CCC2)c(C)cccc1C C1(NC(c2c(CC)n(CC)nc2)=O)COCCN(C(C2(CC)CCCOC2)=O)C1 N1(C(COC)=O)CC(C(=O)NCCn2cncn2)C(F)(F)C1 c1(C(N(CCNC(CC2(C)CC2(F)Cl)=O)C2CC2)=O)ccc(F)c(OC(F)(F)F)c1 c1(OCC)cc(C(=O)NCC2CC(O)(CNC(=O)Cc3ccon3)C2)ccc1C C(=O)(C#CC1(SC)CC1)NCC(CC(C)C)NC(CC(=O)OC)=O C(=O)(CC(C)(C)c1ccccc1)N(C1CC1)CC1N(C(Cc2c(C)con2)=O)CC1 N1(C(C(CC)C(C)C)=O)CCN(C(=O)C(c2cccc(OC)c2)C)CC2(CC2)C1 C12(CNC(C(C)=C3CCC3)=O)CC(CO1)N(C(=O)C(C(C)C)OCC(C)C)C2 c1(NC(c2ccnc(CNCc3cc(B(O)O)co3)c2)=O)cc(Cl)c(Cl)cc1Br C(=O)(C1CC2(CCCC2)C1)N1C2CC(CNC(C3C(C)=CCS3)=O)C1CC2 C(=O)(C(CO)C(F)(F)F)NC1(CC)CCN(C(c2ccc(F)o2)=O)CC1 C1(CNC(C(C(C)C)F)=O)CCC(C)CN1C(C1(n2cccn2)CC1)=O N1(C(COCCCN=[N+]=[N-])=O)CC(C(=O)NC2CC3CCCC3C2)C(F)(F)C1 c1(C(N2CC=CC(NC(COCCOC)=O)C2)=O)ccc2nc(C)nc(O)c2c1 c1(CC(N2C(CN(C(CCCOC)=O)C)CCC2)=O)ccc2nonc2c1 c1(SC)cc(C)c(C(=O)NCC2(F)CCN(C(c3c[nH]nc3C3CC3)=O)C2)o1 Cc1nc(C(=O)NCC2CCCN2C(=O)C(O)CC(C)C)c(C)n1C c1(C(N2CC3CCC2CN3Cc2cc3ccoc3cn2)=O)cc(Cl)c(Cl)nc1Cl CCCC(C)(CC)C(=O)NC1(CCNC(c2cnnc(O)c2)=O)CCC1 c1(CC)c(C(=O)NCC(=O)NCC(N2CCC(C)(CN(C)C)C2)=O)nnn1C N1(C(COCCC=C)=O)CC(NC(C2(CC3CC3)CCCO2)=O)CC(F)C1 C(C(C(C)(C)C)NC(=O)C(c1ccc(Cl)cc1)N(C)C)NC(c1c(C)noc1)=O CC(C)C(CNC(=O)CNS(C)(=O)=O)NC(c1ncc(C(F)F)s1)=O c1(OC)cc(=O)n(C)cc1C(=O)NC(C)CCNC(=O)C(C1CCCC1)OC C(CC(=O)NC1CCS(=O)CC1)(C(F)F)NC(c1cncc(C2CC2)c1)=O C12(NC(c3c(CC)nco3)=O)CCCN(c3cc(C(=O)OC)nc(C)n3)CC1C2 C(=O)(CC(C)CC(=O)N1CC2(CC2)CC1CC(=O)NCC(C)(C)C1CC1)OC c1(NC(Cc2c(N=[N+]=[N-])cccc2)=O)ccc(O)c2ncccc12 c1(C(=O)NC(C)CN(C(=O)CC2(C)CC2)C)ccn(C(=O)OC(C)(C)C)n1 CC(CC(=O)N1CCCC(C(=O)N(C2CC2)Cc2cccs2)C1)CC(C)(C)C C1(O)(C(N2CC3(CC(NC(c4cc(OCC)no4)=O)C3)C2)=O)CCCC(C)CC1 C(CC(C)(C)C)(C(=O)NC(CSC)CC)NC(CCCOCCC)=O c1(C(=O)NC2C=CCN(C(c3occ(C)c3C)=O)C2)ccc2ccccc2c1 c1(CC)ccc(C(=O)NC2CN(Cc3cn(CC4CC4)nn3)CC2F)c(F)c1 c1(C(=O)NCC2C(CNC(c3cc(C)nnc3)=O)C2)cccc2c1ccn2C c1(C(N(C2CN(C(c3c(Cl)cn(CC)n3)=O)CC2O)C)=O)ccn2nncc2c1 C1(C(=O)NCC2CN(C(c3cccc(F)c3)=O)CCO2)CC2CSCC(C1)C2 C1(C(=O)O)CC2(CCCC2)CN1C(=O)C(=O)Nc1cc(F)c(F)cc1F CCC(CNC(c1cnn(C)n1)=O)(CC)C(=O)N1CCCC(CO)C1 c1(CN(C(C(C(=O)OC)CC)=O)C)cc(OC(=O)C(C)(C)SC)cc(O)c1 N1(C(C2C(C)CN(C(=O)C3=C(Cl)CCC3)CC2)=O)CCc2cccnc2C1 C(C(C)C(C)C(=O)N1CCCC1CNC(C1CCOC1C)=O)OC N1(C(c2cn(C)nn2)=O)CCC(NC(c2cc(N)cc(O)n2)=O)C2(CCC2)C1 C(=O)(C(C)(C)CC(=O)NCCc1ocnc1CNC(=O)C(CC)CC)OC C1(C(=O)NC2C3(CCN(C(CS(CC)(=O)=O)=O)CC3)C2)COc2ccccc2O1 c1(C(N(CCOC)CCNC(C2CCC2(F)F)=O)=O)c(C)cc(C)nc1C c1(NC(C23CN(C(=O)CNc4nccs4)C(C2)CO3)=O)ccc2nc(Br)sc2c1 N1(C(c2n(CC)ncc2C)=O)CCC(C(=O)NCCN2CCCC(O)C2)C1(C)C C1(CC(=O)NCC2CN(C(C3OCCC(C)C3)=O)CC2C)CCCC2(CCC2)O1 c1(C(N2CC(N(C(=O)C=CCn3cncn3)C)C(F)C2)=O)sc(Cl)c(Cl)c1N C(C(C)(CC(=O)N(CCCNC(C1CC(N(C)C)C1)=O)CCO)C(F)(F)F)N(C)C Cn1nc(C(C)(C)C)cc1C(c1ccccc1)S(=O)(=O)CC1CCCCN1 C1(CC(=O)NCC=C)CC12CCN(C(=O)Cc1ccco1)CC2 c1(C(=O)NC2CN(C(CC3C(C)(C)CCO3)=O)C2)nc2ccc(Br)cn2c1F C(CS(=O)(=O)c1ccccc1F)NC(=O)NC1C2(CC(OC)C2)C1 C(=O)(C1=NOC(C)(C)C1)NCC1C(NC(Cc2cccc(OCC=C)c2)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)NC(C)CC(C)NC(=O)C(O)CC1CCOCC1 C=CC(C)(C)C(=O)NCC1(CNC(=O)CCSc2csc(C)n2)CCC1 CC1(NC(c2cc(F)cs2)=O)CC(NC(=O)Cc2cncs2)C1 C(=O)(CC(F)(F)CC(=O)OC)N1CCN(C(Cc2ncc(CC)[nH]2)=O)C(CF)C1 c1(C(=O)NC2C(CNC(C3(OC)CCOCC3)=O)COC2)ccc(O)cc1Cl C1(C2CC2)(NC(C2=CC(C)(CC)C2)=O)CCN(C(=O)C(C)(C)C(C)(C)C)C1 CCCC(CC)C(=O)NCC1CCCN(C(c2ccc(C3CC3)nc2C)=O)C1 c1(OC)c(C(N2CC=CC2CNC(C2CC2(F)F)=O)=O)csc1Cl c1(-c2onc(-c3c(C)cc(F)s3)n2)cc2occc2s1 c1(OC)cccc(CCC(=O)N(C2C3CN(C(=O)COC)CC23)C)c1.C(C)(C)N C(C(C)(C)CNC(=O)CCCc1cccnc1)N(C)C(c1nocc1Br)=O C(=O)(C1=CCC(NC(c2ncnc(O)c2F)=O)C1)NC1CCC(C(C)(C)C)C1 c1(CC(C)C)ncc(C(=O)NCC2CCC(NC(C3CC(C(F)F)C3)=O)C2)[nH]1 N1(C(C2N(C(c3c(CC)nccn3)=O)CC(C)C2)=O)CCOC2(CC2)C1 C(CN=c1[nH]c(N2CCN(C3CC3)C(C)C2)nc2c1CCCCCC2)SCC=C C1(NC(c2cn(C(C)C)nc2)=O)CC2CC(NC(=O)C=Cc3ccc(Cl)s3)CC12 c1(C(=O)NCC(=C)C)ccc(CNC(=O)CC2C=CCC2)nc1 CC12CN(C(=O)C(O)C3CC3)CC1CN(C(c1n[nH]cc1Cl)=O)C2 Cc1ccc2n[nH]cc2c1C(N1CCN(C(C2CN(C3CCC3)C2)=O)C(C)C1)=O C1(NC(c2cnc(C(C)=O)s2)=O)CN(Cc2cc(C)sc2C)CC1(C)C N12CC3(CCC1C3)CC(CC)C2=O.n1(CC)cc(CC2(O)CCSC2)nn1 c1(CC)ccc2cc(-n3nc(C4CSC4)nc3C(SC(F)F)C)ccc2c1 C1(NC(c2cc(C3CC3)cs2)=O)CN(C(c2ncoc2Br)=O)CC1O C1(C)(CNC(c2cnc(NC(C)=O)o2)=O)CCN(C(=O)C2=CCCO2)C1 C(CC(C(=O)N1CC=CC1CF)NC(=O)Cc1cccnc1C)SC c1(CC(=O)NC2CCC(C(=O)NCc3csnn3)CC2)ccccc1[N+](=O)[O-] N1(C(Cn2c(=O)sc(C)c2C)=O)CCN(C(=O)C(CO)NC(N)=O)CC(O)C1 C1(C(N2CCC(OCC=C)C2)=O)CCN(C(=O)C(C(C)C)SCC)C(C)(C)C1 n1(CCC)ncc(CNC2CCC(NC(c3cc(Br)ccn3)=O)C2)c1C N1(C(=O)NCCc2sc(C)c(C(C)C)n2)CCOc2cccc(Cl)c21 N1(C(C2(CC)CC(C)(C)C2)=O)CCC2CCC(C1)N2C(=O)CC1(O)CCOCC1 Cc1cc(C(=O)NCC2CN(C)CCN2C(C2COCCO2)=O)cc(F)c1 C1(NC(c2ncn(C)n2)=O)CCCC12CCN(C(=O)CS(=O)(=O)NC1CC1)C2 c1(C(=O)NC(CC)CNC(c2cn(C)nc2CC2CC2)=O)cnc(N)c(CO)c1 C1(CNC(=O)Cn2ncc(Br)n2)CC2(C1)CN(C(C13CCC1C3)=O)C2 c1(CNC(c2ccns2)=O)cn(C2CCCC2)nn1 CCC(C#N)C(=O)NC1CC(NC(=O)CCN2C(=O)CCC2=O)C1 N1(C(C2(CC#C)CCOC2)=O)CC(NC(C2(NC(N)=O)CC2)=O)C(C)C1 C1(CC)(NC(c2scnc2CO)=O)CCN(C(c2nccc(OC)c2O)=O)CC1 C1(CNC(CC2CCN(C)C2=O)=O)CCCC2CN(C(=O)CC3CC3)CC12 CSC=CC(=O)N(C1CN(Cc2cn(C3(C(=O)O)CCC3)nn2)C1)C C1(C(=O)Nc2nc(OCC)oc2)CCN(C(=O)CCOC)C(C)(C)C1 N1(C(C(c2c(C)cc(F)cc2)(F)F)=O)CC2(CCN(C(c3cnc(O)s3)=O)C2)C1 S(=O)(=O)(c1cc(Cl)ccc1OCc1ccccc1)N1CC(CN(C)C)OCC1 CC1(C)COC(CC(N2CC(NC(C3(F)CCCCC3)=O)CC2CO)=O)CO1 C(CCC1CC1)(C(=O)N(C)Cc1cn(C(C)C)nn1)NC(CCSC)=O C1(C(N2C(CCNC(CCCCC)=O)CCCC2)=O)CN2CC3CC2(CO1)C3 C1(CC(=O)N(C2CN(C(=O)Cc3ccccc3)C2)C)CCC12CCC2 C1(C(N2CC(CN(C(CC(C)C)=O)C)OCC2)=O)CCCN(S(N)(=O)=O)C1 c1(C(=O)NCC2CCN(C(C3CC(C)OC3=O)=O)CC2)cc(S(C)(=O)=O)co1 C1(OC)CN(C(=NCc2ccc(F)cc2)NCc2ccc(F)cc2O)CC1OC N1(C(C(=O)NCc2cc(CC)sc2)=O)CCC(S(=O)(=O)CC)C1 c1(CC)ncc(C(N2CCC(NC(=O)CN3C(C)CCC3C)CC2)=O)c(O)n1 c1(C(CC)C)ccc(OC)c(O)c1.C1(C(C)C)(NCO)CC1 Cc1c(C(=O)NCCC2CCCCN2C(C2CC(C3CC3)=NO2)=O)nn(C)c1N c1(C(N2CC(CNC(c3cncc(C)c3)=O)OCC2)=O)nnn2c1COCC2 N1(C(c2cn(CCC)nn2)=O)CC(O)CC1C(=O)NC(C)CCSCC C(=O)(C(C)(C)CC(=O)NCCCN(C(=O)Cc1cc(C(F)(F)F)n[nH]1)C)OC CC1(C)OCCc2cc(C(=O)NCC3CC3NC(c3ccccc3O)=O)ccc21 C1(C(=O)NC(C)(C)CNC(=O)CCC2CNC(=O)N2)CCCC2(CCOCC2)O1 N1(C(C2N(C(c3c(C)n(C)nc3)=O)CCOC2C)=O)CC2(CCC(C)OC2)C1 C1(C(=O)NC2CCC(F)(CNC(=O)C=CC3CC3)C2)CCc2c[nH]nc2C1 N1(C(CN(C(C(C)C)=O)C)=O)CCCC2(CCC(NC(=O)C3=CCCSC3)C2)C1 c1(C(N2CCC(n3cccc3)C2)=O)cc(N2CCC(O)C2)ccc1[N+](=O)[O-] C1(CC(=O)NCC2N(C(C3(COC)CCCC3)=O)CCC2)SC2=NCCN2C1=O c1(CCC)cc(C(=O)NC2COCC2CNC(c2cnc(C)s2)=O)n[nH]1 C(C(CC(C)C)C(=O)NC1CN(C(=O)CN(C)Cc2ccccc2)CC1C)OC c1(C(N2CCCC(C(C)NC(c3cc(C)no3)=O)C2)=O)cn(C)c(=O)cc1C Cc1nc(C)c(CNC(=O)C=CCN(C)C(C2(O)CCOC2)=O)[nH]1 CS(=O)(=O)C(CNC(c1cccc(CO)c1)=O)CNC(c1n[nH]cc1Cl)=O N1(C(C2CCCC2)=O)CCCC(N2CCN(C(C3CC=CCC3)=O)CC2)C1 c1(C(=O)NCC2OCCN(C(C3(CC(C)C)CCC3)=O)C2)cc(N)c(F)cn1 C1(C#CC(=O)NC2CC23CCCC3)(COC)COC1 C(CC(C(=O)NCCCC1(O)CCC1)NC(c1ccc(F)cc1)=O)SC N1(C(CC2CN(C(C)=O)C2)=O)C2CCC1CN(C(C1CC1F)=O)C2 N1(C(=O)CC2CCCCN2C(=O)CC2CCC(=O)N2)CCC2(CC1)CSC2 N1(C(C(F)=CC)=O)CCC(NC(=O)COc2ccc(Br)cc2F)CC1C c1(OC)cc(O)ncc1C(N1CC=CC(NC(=O)CC2CCC(=O)NC2=O)C1)=O C=CCC(C(=O)N1CC=CC1C(=O)N(C(C)CCO)C)OC C12(C(N3CC(NC(CC4CC(OCC)C4)=O)C(C)C3)=O)CCC(CF)(CC1)CC2 c1(C(C)(F)F)cc(C(=O)NCC2(NC(C3CCCC3CF)=O)CCOC2)no1 C12(C(N3CC(C)C(CO)CC3)=O)CCCC1CCN2C(C1CNC(=O)N1)=O N1(C(c2cc(CC)c(O)cc2)=O)CCN(C(=O)CCCC(F)F)C2CCCCC12 C1(C(=O)NCC(CC=C)NC(c2[nH]c(C)c(C(C)=O)c2C)=O)CCCS(=O)(=O)N1 N1(C(CC(C)=C(C)C)=O)CC(NC(=O)C=Cc2ccncn2)CC1C CC(C)CC(CNC(=O)CSCc1ccccn1)NC(=O)CCn1ccnn1 N1(C(Cc2cc(C)on2)=O)CC(C2CCN(C(C3(CCN=[N+]=[N-])CC3)=O)CC2)C1 Cc1cn2cc(CCNC(=O)C(N3CCCC(O)(CN(C)C)C3)=O)nc2s1 c1(C(C(N2C(COC)CC2)=O)C)cn(CC(=O)O)nn1 c1(CCC(=O)NC2C(C)CN(C(CCC)=O)CC2C)c(C)nc2nc[nH]n2c1=O c1(C(=O)NCC2(NC(C(C3CC3)OCC)=O)CCOC2)cc(C)cc(C)c1O C(=O)(C(O)CC(C)(C)C)N(C)CC1CCCCN1C(c1ccnc(Cl)c1N)=O C(C(C(C)C(C)C)NC(=O)Cn1cnc(=N)[nH]1)NC(c1ncn(CC)n1)=O C1(=O)C(C(C)(C)C)N1.C1(NC(C=CC(C)(C)C)=O)COCCC1C(=O)NC(N)=O N1(C(CC)=O)CCC(CNC(=O)CCC2CCCC(=O)N2)C12CC2 C1(NC(C(C)NC(C)=O)=O)CC2CCC1CC2NC(=O)C(C)C(C)O C1(CNC(c2c(CC)ncs2)=O)CC(C)N(C(=O)C(C)Cc2cccc(F)c2)C1 c1(OC(C)=O)cc(C)c(Br)cc1C(N1CC(NC(=O)C=CCO)C(O)C1)=O c1(CCNC(=O)NC(c2ccccc2)CC#C)cc2ccccc2n1C c1(C(N(CCC(N)=O)CC)=O)ccc(CNC(=O)COC2(C)CCCC2)o1 C=CCCC(C)(C)C(=O)N(C)CCOCCCN(C(=O)CCN(C1CCC1)C)C CCC(C)CC(C)N(c1ccccc1OC(F)F)C.C12CCCCN1C2=O n1(C(CC)C)[nH]c(=NC(=O)C=Cc2ccccc2)cc1C c1(C(=O)NC2(C)CN(C(c3cnn(CC(F)F)c3)=O)C2)cnc(O)c(Br)c1 CC(C)(C)CC(F)C(=O)NC(C)(C)CCCC(=O)NC1C=CC(C)(C)CC1 N1(Cc2cc(Cl)cc(OC)c2)CC2CN(C(C3(CF)CC3)=O)CC2C1 C(=O)(C1=CSCS1)N1CC(c2ccccc2)(NC(CCC2N(C)CCC2)=O)C1 CN1CCC(C2CCN(Cc3ccc(-c4nn[nH]n4)o3)C2)C1 C(=O)(CCC(=O)NN(C)C)N(CCC(=O)NCCC1CCN(C)C1=O)CC#C C(CC1CCc2ccccc21)NC(C(=O)NCc1ccccc1OCCF)=O C#CCC(C)(C(=O)Nc1ccc(O)cc1C)NC(=O)C(C)CCCC N1(C(c2oc(C)c(CO)c2)=O)CC2N(C(=O)C(O)CN(C)C)CCC2(C)C1 Cc1ccc(O)c(CNC(=O)C(CCN(C)C)NC(c2cnsn2)=O)n1 C(=O)(C(O)CCCNC(=O)CC1CC2(CCC2)C1)NCCC#CCC c1(C(=O)NC2(C)CCN(C(C3C(=C)C3)=O)C2)ccnc2cc(Cl)ccc12 O=C(C(C1=NOC2CC12)N1CCc2c(Cl)cccc21)NCCC1CC1 CCCCCCCC(=O)NCC1(F)CC(NC(c2ccc(Cl)c(C)c2N)=O)C1 CCS(=O)(=O)CC(=O)N(C)CC1CCCC(NC(=O)COC(=O)CO)C1 C=CC(C)(C)CC(=O)N1CC(C(=O)N(C)CC2CC(F)C2)C(C)(C)C1 Cc1nc(C2CC2)[nH]c1C(=O)NCC1CC(NC(c2c(Cl)cnn2C)=O)C1 c1(C(=O)NC(CSCC)C(=O)NC2CCN(C)C2)cccc(C)n1 Cc1ccc2[nH]nc(-c3nc(Cc4cc(C)sc4C)no3)c2c1 C(C)(C)(CC(=O)N(CCCNC(=O)CC1CCC1(F)F)C1CC1)NC(C)=O C1(C(=O)NCC=CCNC(C2(CC(C)C)CC2)=O)CCCC(F)(F)CC1 n1(CCC)ccc(=NC(=O)C(Cc2ccoc2)NC(=O)CC(C)CC)[nH]1 CC(C)CC(CNC(c1ccc(CO)o1)=O)C(=O)NC(C1CCCC1O)C O=C1CCCC(CC(=O)NCCCCNC(C2CC3CC3C2)=O)N1 C(=O)(CC(C)CN(C)C)NCC1(NC(Cc2scc(C)c2)=O)CCC1 c1(C(=O)NC23CCC(NC(C4CC=C(C)CC4)=O)(CC2)C3)cc(O)cc(Cl)c1Cl C1(C(N2CCC(C)(C)C(CNC(=O)COCCF)C2)=O)Cc2cccc(F)c2O1 Cc1cc(C(N2CCCCC(NC(=O)C=CC3(C)CCOCC3)C2)=O)ncc1F N1(C(C(CC2CCC2)OC)=O)CCCC(C)(C)C1C(=O)NC1COC(C(N)=O)C1 C1(N(C)C(c2coc(O)n2)=O)CCCN(C(c2c[nH]nc2-c2cccs2)=O)CC1 c1(C(=O)NCCN(CCC)C(C2(OC)CCSC2)=O)ccc2c(c1)C(=O)NC2 c1(OC)cc(CC(N2CC3(NC(=O)C(C)OC)CCC2C3)=O)ccc1[N+](=O)[O-] N1(C(C(CC=CCC)C)=O)C2CCC1CN(C(C13CC(C(=O)OC)(C1)C3)=O)C2 C1(C(N2CCN(C(CC(CC)C)=O)C(C)C2)=O)Cc2cccc(OC)c2O1 C1(NC(CNS(CCCC)(=O)=O)=O)CCCN(C(c2c(Cl)n[nH]c2C)=O)CC1F C1(CCC(=O)NC(CC(=O)CCO)C2(C)CC2)(COC)CCCC1.C1(NC)CCC1 N1(C(CCC#C)=O)CCCC(O)(CCNC(=O)C=CI)C1 c1(COC)nocc1NC(=O)C(Cc1cn[nH]c1)NC(=O)C=CC(C)CC S(=O)(=O)(C1CCCCC1)NC1C2CN(c3cc(OC)nc(C)n3)CC21 c1(CC(=O)N(C2CN(C(=O)CNS(C)(=O)=O)C2)C)cc[nH]c(=N)c1 C1(C(=O)Nc2nc(C3CC3)cc(Cl)n2)CCCC12CCN(C(c1ccns1)=O)C2 N1(C(C(C)n2cccn2)=O)CCSCC1CCNC(=O)C(F)=C(C)C N1(C(c2c(CC)cco2)=O)CC2CC(NC(c3nccn3C(C)C)=O)CC(C2)C1 C1(C(N(CC)CC2CCCN(C(=O)CCC=C(C)C)C2)=O)CC2CCC(C1)C2 Cc1ccccc1NCCc1nc(-c2cc[nH]n2)nn1-c1cccc(C(=O)O)c1 C1(C(=O)NC2CN(C(C(C)=O)=O)C(=O)C2)CCC(C)(C)CN1 C1(NCCc2c(OCC)nccc2)CC2CCC1N(C(=O)OC(C)(C)C)C2 CC1CC2CN(C(=O)CC(Cl)Cl)CC2N1C(c1cscc1Cl)=O c1(CC(=O)N(CC(CNC(C(C(C)C)F)=O)O)C)csc2ccc(Cl)cc12 C12(C(N3CCC(C)(N(C)C)C3)=O)CC(CN(C(C3CCCCCC3)=O)C1)C2 c1(OC)ccc2c(c1C(=O)NC1CCN1C(=O)CC(C)C1(OC)CCC1)CCC2 C(=O)(C=C1SCC(=O)N1C)NCCC1=CCN(C(C=C2CCC(C)C2)=O)CC1 Cc1nn(C)c(C)c1C1CC(C(=O)OCCCc2ccc(N)cc2)CCO1 CC(C)(C)CCCNC(c1sccc1CNC(=O)CCCC1CCC1)=O N1(C(c2c(C)nc(O)cc2)=O)CCC2(CC(NC(C3(C)CCC3)=O)CO2)C1 C1(C(N2CCCC(CNC(C3=CCCC3C)=O)(CO)C2)=O)CCc2nnnn2C1 c1(CC(=O)NC(C)CC(C)NC(C2(O)CC2)=O)ncc(F)cc1F N1(C(C2(OCC)CCC2)=O)CCC(CNC(=O)Cn2ncn(C)c2=O)CC1 Cc1nc(O)c(Br)cc1C(N1CC2C(NC(=O)C(C3CC3)N(C)C)C2C1)=O C1(C(=O)NCC2(F)CN(C(C(C)(C)OC(C)C)=O)C2)CCC12CCCO2 C1(CNC(C(C(=O)OC(C)(C)C)(C)C)=O)CN(C(=O)C(F)F)CC2(CCC2)O1 C1(C(N2CCCC(NC(Cc3c(C)ccs3)=O)C2C)=O)CC2C=CC1CCC2 c1(C(=O)OCC)c[nH]nc1S(=O)(=O)NC1CCN(c2ncccc2Cl)CC1OC N1(C(C2C(C(C)C)OCC2)=O)C2CCC1CC(N(C)C(C13C=CC(CC1)C3)=O)C2 C(C)(C(=O)NCCC1(C(=O)NCC2CCCO2)CCC1)=C(C)C C(C(C)(C)CC(=O)OCc1ccccc1CCCN(C1CC1)C(C)C)OC CS(=O)c1ccccc1C(=O)NC1CC12CCN(C(C1C3CCC1CC3)=O)CC2 c1(CC(N2CC(C(C)NC(c3ccnnc3)=O)C2)=O)nn(C)cc1[N+](=O)[O-] c1(C(=O)NC2CC(CCNC(c3c(OC)scc3)=O)C2)cccc(S(C)=O)c1 c1(C(N2CC3(CCN(C(Cc4c(C)noc4)=O)C3)C2)=O)cc2c(cn1)OCCC2 N1(C(C(C2N(C(c3cncc(C)n3)=O)CCC2)(C)C)=O)CC2(CCOC2)C1 c1(C(N2CC(OC)C(NC(=O)C(C)NC(C)=O)C2)=O)ccc(S(C)(=O)=O)c(C)c1 N#Cc1cnc(NC2CC2)c(Br)c1.C12N(CC13CCCC3)C2=O Cc1nc(CC(=O)NCC(C(C)(C)C)NC(c2csnc2Br)=O)c(C)s1 C(=O)(C(O)C(F)(F)F)N(CCN(C)C(c1cccc(C(C)(F)F)n1)=O)C Cc1nc(=N)[nH]cc1C(=O)NC1CC1NC(c1cnc(C(C)(C)C)nc1)=O Cc1cccc(COCC(=O)NC(c2ccc(CNC(=O)C(C)O)cc2)C)c1 CC1CN(C(c2cn(CCNC(c3cc(O)cc(=O)o3)=O)nn2)=O)CC(C)(C)C1 Cn1cncc(C(N2CCC(NC(=O)CN3CCCS3(=O)=O)C(F)C2)=O)c1=O C1(CC(=O)NCCN(C(=O)CC2SC(=N)NC2=O)C)COC(C)(C)C1 c1(OCC)c(C(C)NCC2CC23CCOCC3)c(C)nn1C C(=O)(CC1CN(C(c2cc(C)c(C)n2C)=O)c2ccccc21)OC C(=O)(C1=NN(C2CC2)C(=O)CCC1)N1CCC(C)(CNC(CC(C)F)=O)CC1 c1(C(=O)NC2CC(C)(CNC(CSCCN(C)C)=O)C2)cnc2n1CCC2 C1(SCC(=O)Nc2c(N(C)C)cc(C)c(Cl)c2)Cc2ccccc2CN1C C1(C(=O)NCCC#CCC)C2CCCC2CN1C(=O)CCCOC Cc1ccc(C(N2CCCC(C)C2CNC(c2cnoc2C)=O)=O)c2c1CCC2 CN1CCc2cc(C(N3CCC4(NC(CSCC(C)C)=O)C(CC3)C4)=O)ccc21 c1(OC)cc(C(=O)NCCC(N2CCCCCC2)C)cc([N+](=O)[O-])c1 N1(C(C(CC)C(C)O)=O)CCN(C(=O)CCOc2c(C)cccc2C)CCC1C CC1CCC(CNC(c2cc[nH]c(=N)n2)=O)CN1C(=O)C(C)Oc1ccccc1 C1(C(N2CC(N(C(=O)CCC3CCC(=O)N3)C)C2)=O)CC12CC(O)C2 c1(OC)ccc(C(=O)N(C)CC2CN(C(=O)C(C)C#N)CCO2)c(C)c1 c1(C(C)=O)ccc(C(=O)NCC=CCNC(=O)C(C)Oc2ccccc2Cl)nc1 CC1C(NC(C2CCC(F)(F)C2)=O)CCN1C(=O)CCCC1CCCC1 N1(C(=O)O)CCC(C(=O)OC(C)(C)C)CC1C.c1(C(=O)OCC)ncn(CC)n1 CC(C)C(CNC(=O)CN1CCCC1=O)C(=O)NC1C=CCCC1 C1(C)(C(N2CC(C(N)=O)(CNC(CNS(CCOC)(=O)=O)=O)C2)=O)CCC(C)C1 N1(C(=O)Nc2ccc(C)o2)CC(NC(=O)CC2CCCCO2)C(C2CC2)C1 N1(C(Cc2nc(C)c(C)s2)=O)CCC2(CC1)CC2NC(c1ccc(F)c(F)c1)=O N1(C(c2c(=N)[nH]cnc2)=O)CCN(C(=O)COCc2ccccc2)C2CCC12 N1(C(C(CC)C2CCOCC2)=O)CCC(CC=C)(NC(C2CCCSC2)=O)CC1 c1(C(N2CCC(C3(C)NC(=O)NC3=O)CC2)=O)n[nH]c2cc(N)ccc12 C1(OCC(F)(F)F)CCCN(Cc2ccc(F)cc2C(F)F)CC1 c1(C(N(C(CC(=O)NC2(CC=C)CCOC2)C)C)=O)c(Cl)cnn1CC C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)N(C(c1ccc(N2CCOCC2)cc1)=O)CC C(CCCCCC(=O)NCCc1nc(C2CC2)n[nH]1)NC(C(CC=CC)C)=O Cc1ccc(CC(=O)NCC2CCN2C(C2CCOC2C(C)C)=O)cc1C CC(C(C)(C)C(=O)NCC12CCN(CC1)C2)NC(=O)C(C)N=[N+]=[N-] C(N=c1[nH]c(Cl)c(C#N)s1)C1OCCCN(C(c2n(C)c(O)nc2)=O)C1 C(C1=NOC2CN(C(C3CC(O)C3)=O)CC12)NC(c1c(CC#N)cccc1)=O Cc1ccc(C#N)c(NC2(CO)CCN(C(=O)CSc3cccs3)CC2)n1 c1(C(=O)NC2CCC(N(C)C(C3CC4CCC3O4)=O)CC2)cccc2cnnn12 N1(C(c2nc(C)oc2)=O)CC2(C(N3CCC(C(F)F)C3)=O)CCC1CC2 CCC(C)(C(=O)N1CC2CC1C2NC(c1cc(Cl)c(F)cc1F)=O)C(N)=O C1(C(=O)NCCCC(CCC)NC(c2cccn2C)=O)CCC2(C1)CC2(F)F Cc1noc(Cl)c1CC(=O)N(CCNC(=O)CC1CCCC(O)C1)CC1CC1 C1(COC)CN(C(=O)NC2CCOC(c3cncn3C)C2)CCC1(F)F C(=O)(CCCCC(C)C)NCC(CNC(c1c(OC)ncnc1OC)=O)(C)O c1(C(=O)NCCN(C(Cc2c(SC)cccc2)=O)CC(C)O)ccc(N)c(F)n1 c1(-c2cc(OC)c(C)cc2)n[nH]c2ncc(C(=O)NCCSC)cc12 N(C(=NCCCCl)NC1CCCN(Cc2ccccc2)C1)CC(N(OC)C)=O C1(C(=O)NC2CC(Cl)(Cl)C2)CC(O)CN1C(=O)Cc1cnns1 C=CCCCCCC(=O)N(CC(C)O)CCNC(c1cnc(NC(C)=O)o1)=O C1(CC(=O)NCCC2(NC(c3cc(C)no3)=O)CC2)OCCOC1(C)C c1(NC(C2CCC(NCc3ncc(C)s3)C2)=O)ccc(Cl)cc1F Cc1cnc(C(C)NC(=O)C(C2CCCCN2)c2ccc(Br)s2)s1 C(=O)(C(F)(CNC(C1CC2CCC2C1)=O)C(C)C)NCC(C1CCCC1)OC C(C(CC(F)(F)F)NC(=O)C(C)COC)NC(c1cnc(OCC)s1)=O Cc1cc(C(=O)NC(Cn2cncn2)C(=O)Nc2cccc(O)c2)nn1C C1(NC(c2nc(CCCC)sc2)=O)CS(=O)(=O)CC1NC(=O)C1CC1 N1(C(C2C(CNC(Cc3n(C)cnn3)=O)CC2)=O)CCOC2(CCC2)C1 c1(C(=O)NC(CNC(C2CC(C(C)C)C2)=O)(C)CC(C)C)cc(F)cc(Cl)c1N c1(C(=O)NCC23N(C(CNC(=O)NC)=O)CC(C2)C3)c(C)cc(OC)cc1F c1(-n2c(CCC)nc(-c3occc3C)n2)ccc(C(=O)OC)c(C)c1 c1(C(N2CCCC(N(C(C(=O)NCC)=O)C)C2)=O)c(SC)nc(O)nc1C C1(C(=O)NCc2occ(C(N3C(C)(CCC)CC3)=O)n2)CC2CC1CC2=O c1(C(=O)NC2(C)CC(NC(C(C)OC)=O)C2)ccc(Oc2ccc(F)cc2)cc1 N1(C(c2c(CC)[nH]cc2)=O)CCCN(C(C2CC3C=CC2CC3)=O)CC1C Cn1cc(Cl)cc1C(=O)NCC(=C1CN(C(c2cnnc(C3CC3)c2)=O)C1)F C1(C(=O)NC(C)CN2CCCCC2)CCN(C(=O)Cc2ccn(C)n2)C(C)C1 C12(CC(N3C(C)CC(NC(CCCC(C)=O)=O)C3)=O)CCC(CC1)C2(C)C N1(C(COCCC#C)=O)CC2CN(C(=O)Cc3ccnc(O)c3Br)CC2C1 C1(O)(C(=O)NC2(COC)CCN(C(C3CCSC3)=O)CC2)CCCC(C)(C)CC1 C(=O)(C(O)Cc1cnc[nH]1)NCC(CC)N(C(=O)CC(C)n1ccnc1)C Cc1ccc(OCCC(C(=O)CS(=O)Cc2nonc2C(=O)O)=O)c(C)c1 CCC(CC(=O)NCC(C)(CC)NC(c1ccc(OC)cc1OC)=O)C(C)C C12(C(N3CCC(C)CC3)=O)COCC1CN(Cc1ccc(O)c(I)c1)C2 O=C(CC1=CCN(C(=O)C(F)CC2CCOC2)CC1)NCC(c1cnn[nH]1)O CC(F)CN=C(NCc1csc(C(F)(F)F)c1)NCc1ccnn1C CC1(C)COC(=O)C1.C1(NC(=O)OC(C)(C)C)CCCCS1 N1(C(=O)Cn2cccc2)CCN(C(c2cnn[nH]2)=O)C2CCCCC2C1 c1(C(=O)NCC(CN(C(C2(CCOC)CCC2)=O)C)O)ccc(C)o1 N1(C(c2cc(COCC)on2)=O)CC(CC(N2CC=CCC2)=O)C2(CC2)C1 C1(CNC(c2snc(O)c2Cl)=O)C2CN(C(C3(CO)CC3)=O)CC12 C=CC(C)(CCOC)C(=O)N1CCC(O)(CCNC(C2CC2COC)=O)CC1 N1(C(C(CC)(C)O)=O)CCOC2(CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)C1 N1(C(c2c(CC)ncnc2)=O)CCC=C(C(=O)NCC(O)CN(C)C)C1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(NC(c2cn(C(C)C)nc2C)=O)CC1C N1(C(CC(C=C)C)=O)CCC(NC(c2ccc(F)o2)=O)C(O)C1 c1(C(=O)NC(CNC(C(C(C)O)NC(C)=O)=O)(C)C2CC2)cc2c([nH]1)CCCC2 Cc1nnc(C(C)NC(c2conc2C(C)NC(c2ccoc2Cl)=O)=O)s1 CN1CCCC1C1CCCN1C(c1cnc(-c2cnn(C)c2)cn1)=O S(=O)(=O)(c1ccc(NCCC2CC2(Cl)Cl)c(Cl)c1)NCC1(C)CC=CC1 C(=O)(C(CCC(N)=O)n1cc(-c2cccc(Cl)c2F)nn1)NCC1(S(C)=O)CC1 CCCC(C(O)C(=O)NCC(F)F)NC(=O)Cc1cccnc1 C(=O)(CCCCCC(C)C)NCC1N(C(C=CC=CCC)=O)CC(OC)C1 C1(NC(CCC2(C)CN(C(C3CC3[N+](=O)[O-])=O)C2)=O)CCC=CCCC1 C1(C(N2C3CC(CCNC(CN(C)C)=O)CC2CC3)=O)CCCCN1S(N)(=O)=O CCC(CC)C(C)C(=O)N(CCNC(C1CC1C1CCC1)=O)Cc1ccccc1 CC(C)CC(CNC(=O)CC1CCC(C#N)C1)C(=O)NC1CNC(=O)C1 Cc1ncn(C)c(=O)c1C(=O)N(C(CNC(c1cnc(C)n1C)=O)C1CC1)C C1(C(N2CC(O)(C(C(=O)NC(C)(C)C)F)C2)=O)CC12CCCC2 Cc1cc(F)c2cc(C(N3CC(NC(=O)CCN(C)C)C(O)C3)=O)[nH]c2c1 n1(CC)ccc(C(=O)NCC2(NC(=O)CCOCCN(C)C)CCCCC2)c1C N1(C(C23CCC(NC(CCS(CC)=O)=O)(CC2)CC3)=O)CCCC2CCCCC12 Cn1ccc2ccc(C(N3CCC(NC(C4CC(C#N)C4)=O)C3)=O)cc12 N1(C(C(C)C2(O)CCC2)=O)CCC(NC(=O)C(O)c2ccsc2)C1 C#CC1(O)CCN(C(C2CC3CCC(C2)N3C(=O)CC2CCN(C)CC2)=O)CC1 C1(C(C)C)CN(C(=O)CC2CCCN2C(C23CCC(C2)C3)=O)CCO1 C1(NC(c2ccc(OC)o2)=O)CC2CCC1(C(N1CCCN(C)CC1)=O)C2 N1(C(CCN(CCC)C)=O)CCCC(C(C)C(=O)N2CC(CC(F)F)C2)C1 c1(OC)cc(Br)cc2c1C(NC(C13CCC(CC1)CC3)C)CO2 N1(C(C(C=C)O)=O)CCC(N(C(=O)CC2CCCCC2)C)CC1 N#Cc1cc(CNC(=O)Nc2ccc3c(c2)CCCC3)cc(F)c1 N1(C(c2c(CSC)cccn2)=O)CC2CCCC2(CNC(=O)C(Cl)=CCl)C1 C1(CNC(c2ccc(CNC(C3(C)CCOC3)=O)s2)=O)CC2CCC1CC2 C1(CN(C)C(C2(C)CCOC2)=O)CCCCN1C(=O)Cc1cscc1Br c1(OC(C(=O)NCC(C)(C)NC(c2cnc(Cl)[nH]2)=O)(C)C)ccc(Cl)cc1 C1(C(=O)NC2CCC(NC(c3coc(O)n3)=O)CC2)CC2CCCCCCC12 c1(C(=O)NCC(C2CC2)NC(CC2CC(C)C2)=O)cc(-c2ccncc2)[nH]n1 N1(C(C(c2cccc(C)c2)F)=O)CC2(CCN(C(=O)CC3CCCO3)C2)C1 Cn1nc2c(c1C(N1CCC(CC3CN(C(=O)C(F)F)C3)CC1)=O)CCC2 C1(CCOC)CN(C(c2ccc(OC)s2)=O)CCN1C(C1CS(=O)(=O)C1)=O C(CN=c1ncc(F)c[nH]1)C1CC(O)(C(F)F)C1 N1(C(C(N2CCOCC2)C)=O)CCC(N(C(=O)CCC2CCCC(=O)N2)C)CC1 C1(C#N)(CO)CCCOC1.C12CCN(CC1)C(=O)C1CCC(CC1)N(CC)C2 C(=O)(C1=NOC2(CCCN(C(c3cc4ccccc4[nH]3)=O)C2)C1)NC(C#C)C N1(c2cc(C)[nH]n2)CCN(C(C(=O)NC2CCOC2)C2CC2)CC1 C1(NC(CCC2C(C)=NNC2=O)=O)CCC(O)CN(C(=O)CC(F)(F)Cl)C1 CCC(C)C(O)CC(=O)N1CC=C(C(=O)N(C)CCN2CCCC2)CC1 C1(NC(CCC)=O)CCN(C(=O)CC(C)(C)C#N)CC1CO c1(NC(C(=O)NCC(CCCC)CC)C)ccc2c(c1)C(=O)NCCC2 C#Cc1cccc(C(N2CCN(C(C3CC(C)=NO3)=O)CC2C2CC2)=O)c1F c1(C(=O)OCC=C)cccc(OCC2C3CN(C(=O)COCCOC)CC23)c1 C1(NC(C(CCSC)O)=O)(CO)CCN(C(c2cccc(Cl)c2Cl)=O)CC1 O=S1(=O)CCCC(CN2CC(CCCn3cc(CN4CC5CC5C4)nn3)C2)C1 C1(C(=O)NCC2CCCN(C(=O)Cn3cnnn3)CC2)C2CCN(CC2)S1(=O)=O CCCC(CCC)CC(=O)N1CC(n2cc(COC3COCCN3)nn2)C(C)C1 C#CCCCC(C)C(=O)N1CC(CNC(C2CCS(=O)(=O)CC2)=O)OC(C)(C)C1 c1(C(=O)NC2(C)CCN(C(c3c(C)nc[nH]3)=O)CC2)cc(Cl)c(F)cc1F N1(C(c2c(=N)[nH][nH]c2)=O)CCC2(CCCN(C(C3CSCCS3)=O)C2)C1 C1(NC(CC)=O)CCCN(c2nnc(C3CC3)n2CCC#N)C1 c1(C(=O)NC2CC(CNC(CN3C(C)CCC3C)=O)C2)ccc2n[nH]cc2c1 c1(CC(=O)NCC(C)NC(COc2ccc(C)cc2F)=O)c(C)cc(C)cc1C CC(C)C(O)C(C)C(=O)N(CC(N1CCCC(F)(F)C1)=O)CC1CC1 CC(C)C(F)(CNC(C1CC1[N+](=O)[O-])=O)C(=O)Nc1cc(C#N)ccc1O c1(C(=O)NCCCC(C)NC(=O)C(C)(C)Cc2cnn[nH]2)cc(Cl)ccc1Cl c1(C(N2CCC(NC(CC=C=C)=O)C2)=O)cc2nc(CC)cc(C(F)F)n2n1 CC1(C)CN(C(=O)CCC#N)CCN(C(C2CCC3(CCC3)O2)=O)C1 C1(C(N(CC(CO)(CO)NC(C(CSC)C)=O)C)=O)CCC2CCC(=O)N12 C1(NC(c2cc(OC)ns2)=O)CCN(C(c2ccnc(O)c2)=O)C(C)C1 c1(CC(=O)N(C(CNC(CCOCC)=O)C2CC2)C)cc2ccccc2c(=O)o1 C1(NC(C2ON=C(C)C2)=O)CN(C(=O)CCCc2nnc(C)n2C)CC1C c1(C(=O)NC2CC(C)N(C(C3COCCOC3)=O)CC2)cncc2ccccc12 c1(N2CCCC(CCCC)C2)ccc(S(=O)(=O)NC2CCCC2)cc1C#N O=C1NC2(CCCC2)C(=O)N1Cc1nnc(-c2c(Cl)cccc2Cl)o1 O=C1CC(CNC(=O)C(Cc2cnc[nH]2)NC(=O)COc2ccccc2)CCN1 c1(C(N)=O)ccc(Cl)c(NC(=O)C(N2CCCC(C)(c3cccnc3)C2)=O)c1 N1(C(=O)C=Cc2ccoc2)CC2(CCC(C(N3CCC4(CCCN4)C3)=O)O2)C1 c1(C(=O)NCCCCCCNC(C2C3C4CCC(C4)C23)=O)cc2c(o1)CCCC2 C1(C(N2CCC(CN=c3[nH]nc(CCC)s3)CC2)=O)C(O)C(=O)N(C)C1C N1(CC)CCCC(C(N(Cc2ncc(N(C)C)s2)Cc2ccc(OC)cn2)=O)C1 C(CF)(C(F)(F)F)NC(C1C=CCN1C(C1CC1(F)Cl)=O)=O C=C=CCCC(=O)NCc1cc(C(=O)NCCC(O)C2CCCC2)co1 C1(NC(c2cc(O)ncn2)=O)CCC2(CC1)CN(C(=O)CC1CCSC1)C2 C1(C(N2CCN(C(C#C)C)CC2)=O)CCCC(NC(c2csc(O)n2)=O)CC1 C(=O)(C1CSc2ccccc21)N1C2CC(CNC(C(C(C)(C)O)(F)F)=O)(OC2)C1 N1(C(CN(S)C)=O)C(Cn2cc(-c3nccs3)nn2)CC2CCCC12 N1(C(c2cc(C)n(C)c2C)=O)CCC(C)(C)C(CNC(=O)CC2CC=CCC2)C1 C1(NC(C2C(C(N)=O)C2)=O)CC12CC(NC(c1ccncc1)=O)C2 CC(CC#N)C(=O)NC(C(=O)NCCOC1(C)CCC1)C1CC1 N1(C(CC2(CC)CCC2)=O)CC(O)CC1(C)C(N1CCC(CC(C)C)CC1)=O C1(CC)CCC(C(=O)N(C2CCCCC2)CCCNC(C2CCO2)=O)O1 c1(C(=O)NC(C)CC2CN(C(=O)Cc3ccon3)C2)c2n(c(=O)n1C)CCCC2 C(N=c1[nH]c(=NC2C=CC(C)(C)CC2)c2[nH]ccc2[nH]1)c1cncc(OC)c1 CC(C)CC(C(=O)NCCCCNC(c1cccnc1F)=O)C(N)=O N1(S(c2ccc(C(N)=O)o2)(=O)=O)CCCCCCCCCCCC1 c1(CC(=O)NCC(CNC(C=CC(C)=O)=O)O)cccc(F)c1F c1(C(=O)N(c2ncc3ccsc3n2)CC2CCNC2)cc(Br)ccc1[N+](=O)[O-] C1(NC(C2CC=CCC2)=O)CC2(CCC(CNC(C3(c4cc[nH]n4)CC3)=O)OC2)C1 C(CCN=c1[nH]c(=NCC(CC)(CC)C(N)=O)[nH]c2cc[nH]c12)OC=C N1(C(CN(C)CC)=O)CCCC(CN(C(=O)CC2(C)CC2(F)Cl)CC)C1 CC(CCCC(=O)NCC(F)(F)C1CC1)NC(C1CC(=O)N(C)C1)=O c1(-c2ccc(NC(c3cc(Br)cnc3F)=O)cn2)ccc(F)c(O)c1F C(C1CCC(C)CC1)=C(C)C(N1CCCC1CN(C)C(c1cccc(Br)c1)=O)=O C1(C)(C(N2C3CN(C(c4cc(C)nc(O)n4)=O)CC2C3)=O)CCC2(CC1)CC2 C1(C(=O)NCC(C(C)C)C(C)C)CC2C=CC1N(C(=O)C(c1cnn(C)c1)=O)C2 C#CCCCC(=O)NCC1(O)CCN(C(c2ccc(COC)cc2)=O)C1 c1(CC)ccc(C(=O)NC2CC2CNC(=O)C(CCSC)NC(N)=O)c(F)c1 CC(CCl)(CCl)CS(=O)(=O)NCc1ccc(N2CCCS2(=O)=O)cc1 C(CC(=O)NCC(C)N(C(=O)C(C)c1cc[nH]n1)C)SC N1(C(Cn2ccc(C(=O)OC)n2)=O)CCC2CC2(NC(C2CC3CC3C2)=O)CC1 c1(C(N2CCN(C(c3c(OC)csc3)=O)CC(O)C2)=O)c(C)nc2ncccn12 c1(C(=O)NCC(CCNC(=O)CCc2nc[nH]n2)OC)cccc(O)c1 c1(N(CCNC(C2(C3CCCO3)CC2)=O)CC)cc(C(F)(F)F)nc(CC)n1 C(=O)(C1=NOC(C)C1)NC(CC=C)CNC(=O)CCc1ccc(O)cc1 N=c1nc(N2CCOCC2C2CCOC2)c(I)c[nH]1 c1(NCC(CC(C)C)OC)cc(N(C)Cc2cccc(F)c2C)nc(COC)n1 N1(C(=O)CN2CCOCC2)CC2CCN(C(=O)CCc3ccc(Br)cc3)C2C1 C1(NC(c2ccc(C(N)=O)s2)=O)(CO)CCCN(C(=O)CC2CC3CC3C2)C1 c1(CSCC)ccc2oncc2c1.N12C3CCC1(CC3)CNC(=O)C1(CC1)C2=O C(=O)(CCCC(=O)NC1COCC1NC(=O)CN1CC(=O)NC1=O)OCC n1(CC)nc(CNC(=O)C(C2CCC(F)(F)C2)O)c(Br)n1 C1(C(=O)NC2CN(C(C(CCC)CCC)=O)CC2COC)CCc2ccccc2O1 C(CC(=O)N(C1CN(C2CC2)C1)CC1CC1)N(C(C1(CCC=C)CC1)=O)C CC(C)CCCCCC(=O)N(CC(=O)N(c1ccoc1)C)CC(C)C c1(C=O)ccc(C(C)O)cc1.c1(COCC)cn(CC2CCC(C(=O)OC)C2)nn1 C1(CC(=O)NC(C)CCC=C(C)C)(OC)CN(C(=O)CCc2cccnc2)C1 c1(OC)ccc(C(=O)NCCN(C)C(C2(c3ccncc3F)CC2)=O)c(N)c1 C1(CNC(CCCC)=O)CN(C(=O)CC(CC)SC)CCC12CCOCC2 Cc1ccc(F)c(C(=O)NCC2C(C)CCCN2C(=O)CC2COCCO2)c1 c1(N(C)CCN2CC=CCC2)nnc(C=C2Cc3sccc3C2C)n1CCC#N c1(OCC(=O)NC2C(NC(CNCc3cn(C)nc3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 N1(C(C2(C)CCCS2)=O)CCOC(CCCNC(C2(CO)CCCO2)=O)C1 N1(C(C=CC=CC)=O)CCCC(F)(C(=O)NC2(C3CCCC3)CC2)C1 Cc1c(NC(=O)NC(c2cn(C3CC3)nn2)(C)C)oc2c1ccc1ccccc21 C(C1=NOCC1)(C1CCCCC1)NC(C=C)(C)C1CC1 C(=O)(C(CC(C)C)C(C)C)N1CC(CC)N(C(c2sccc2OC)=O)CC1 CC1(C)CC(NC(C2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)=O)C(=O)O1 Cc1ccnc(O)c1C(=O)NC1CCCC(NC(C2CC3(CCCC3)C2)=O)C1 O=C1OCC(COC(c2cn(-c3ccccc3)nn2)=O)O1 c1(C(=O)Nc2nnc(CN(C)C)s2)coc2c1C(O)CCC2 N(C(=NCCF)NC)Cc1cn(-c2ccccc2F)nn1.C(CN(C)C)(C1CC1)OC N(C(=NCCS(=O)(=O)C1CCOCC1)NCC1CC12CC2)CC1CCS(=O)(=O)C1 C(c1cn(C)nn1)=CC(=O)NC(C(=O)NCCCCN(CC)CC)CC1CC1 N1(C(C2CC3(CC(NC(C(CSC)C)=O)C3)C2)=O)CCC(C)C2(CCC2)C1 C=CC(C)(CCOC)C(=O)N1CC(N(C)C(c2csc(O)n2)=O)C1 c1(C(N(C)CCN2CCN(CC(=O)O)CC2)=O)ncnc2c1c(Br)cn2C c1(NC(c2ccc(OC(F)(F)F)c(Cl)c2)=O)cc(F)cc(Br)c1Br C1(C(=O)OC)CCN(c2nnc(CO)n2CC2CCOC2)CC12CCC2 N1(C(C(C=C)O)=O)CCn2ncc(CNC(=O)C(n3ccnc3C)C)c2C1 CC1(C)CCC(C(=O)N(CC(N2CC3(CCC3O)C2)=O)C2CCC2)CO1 C#CC1CCN(C(C23CC2CN(C(C2CCCN2C)=O)C3)=O)CC1 C12(CNC(Cc3cn(CC)nn3)=O)CC(CNC(=O)C(C)NC(N)=O)(CO1)C2 c1(C(=O)NC(C2(C(=O)NCC3CCC4CC34)CC2)C)n[nH]c2ccccc12 C1(C(N(CCCN(C)C(C2CC2(Cl)Cl)=O)C)=O)OCC1(C)C C1(C(N(CC(=O)NCC(F)Cl)CC)=O)COCCN1CC N1(C(c2cccc(OC)c2Cl)=O)CCC2(CCCC2NC(=O)CSC2CC2)C1 CC(O)CCCN(CC(C)N(C)C)CCNC(C1CCCO1)=O C1(c2nnc(CCNC(CC)=O)s2)CCN(C(=O)C(CC)C2CCCO2)CC1 c1(CC(=O)NC2C(CNC(C(COC)(F)F)=O)C2)ccc(OC)c(F)c1.OC CCCC(C)(O)CC(=O)NCC1CC(NC(c2cc(Br)cn2CC)=O)C1 N1(C(CCOCCOC(C)=O)=O)CCC(O)(CN(C(=O)C(C)NC2CCC2)C)C1 Cc1n[nH]c2cc(C(=O)NC(CNC(=O)C3=CCC3)C(C)C(C)C)ncc12 C1(C(N(CCC(C)NC(=O)CCCCC(C)(C)C)C)=O)COc2ccccc2O1 C1(C(N2CC(NC(C3N(C)CCC3)=O)(CO)C2)=O)CC2COCC(C1)C2=O CC1CCN(C(=O)CC2(NC(C3CC(=O)CCO3)=O)CCC2)CC1O N1(C(C(c2scc(C)n2)(F)F)=O)CCC(C2CCN(C(C3C(C)C3C)=O)CC2)C1 c1(NC(C(CNC(C)=O)(C)C)=O)c(C)cc([N+](=O)[O-])cc1Br C=CC(CCC)CC(=O)N1CCC2CC12C(=O)N(C)CC1CCN(CC)C1 Cc1nccc(CNC(=O)CC(C2CC2)NC(=O)CN2CCCCC2C)n1 CN1CCCC(C(=O)NC2CN(C(C3(C#N)CCCO3)=O)CC2F)C1 c1(CC)nc(CNC(=O)C(C2(C)CC2)NC(c2cocn2)=O)co1 C1(CCNC(c2scc(C)c2C)=O)CCCN(C(C2CC3(CCCO3)C2)=O)CC1 C1(CC=C)(C(=O)N(C)CCO)CCN(C(=O)CC2(O)CCCC2)CC1 c1(CC(=O)NCC2CCC(NC(=O)Cc3nocc3Br)C2)ccccc1CCO Cc1cnnc(O)c1C(N1CCC(CNC(C2(CCN(C)C)CC2)=O)C(C)C1)=O Nc1ccc(Br)c(C(=O)NCCCNC(=O)C=C2CC2)c1 Cc1cc(=O)n(C)cc1N1CCN(CC(N2CCCC3(C2)CNC3)=O)CC1 Cc1cc(CCC(N2CC(C)(NC(c3cc(C(F)F)ncn3)=O)C2)=O)c(C)s1 C1(NC(C2CN3CCC2C3)=O)CCCCC1C(N1CC(CCO)C1)=O C1(NC(c2ccc(OC)s2)=O)CCC2(C1)CN(C(c1ccc(F)c(F)c1C)=O)C2 C1(CCC#C)CCCN(C(=O)C(C)CC=CCCNC(C2(SC)CC(=O)C2)=O)C1 C1(CNC(CC(CC)SC)=O)CC(C)(C)CN1C(c1cnn2ccsc12)=O c1(CNC(C(C(C)C)(C)C)=O)ccc2c(c1)CN(C(=O)C(O)Cc1ccccc1)C2 C(C(C(C)C(C)C)NC(c1ccoc1C1CC1)=O)NC(C1(CCCC)CC1)=O c1(NC(C(=O)NC(CCN(C)C)(C)C)=O)ccc(F)cc1C(F)(F)F C1(C(N2CC(CNC(=O)COCC3CCCC3)C2)=O)OC2CCC1CC2 C#CC1(C(=O)NC(c2cccc(C)n2)C)CCN(C(c2cc(C3CC3)no2)=O)C1 c1(C(C)C)ccc(C(=O)NC2CCN(C(=O)Cn3cccc3)CC2CO)cc1Cl C1(N(C(C(C)NC(c2cc(OCC)c(F)cc2)C)=O)C)CCc2ccsc2C1 c1(C(N2C(CNC(CC3(CN(C)C)COC3)=O)CC2)=O)ccc(Br)cn1.CCO C1(C)(CNC(C(N2CCCOCC2)C)=O)CN(C(=O)C(F)C(F)(F)F)C(C)(C)C1 C(=O)(C1=CC2(CCOC2)C1)N(CC(C)NC(c1cccc2cccn12)=O)C c1(C(c2n(CCSC)nnn2)Nc2ccc(-c3ccco3)cc2)cnccc1C c1(C(N(CC(CNC(CCc2cc(C)on2)=O)(C)C)C)=O)cnn(C)c1C N1(Cc2nnc(C(C)C)s2)CCC(NC(c2cc(O)nc(O)n2)=O)C(C)C1 C(=O)(C(O)C1=CCCCC1)N(C)CCNC(c1ccnc(C(F)F)c1)=O C(=O)(C1=NOC(C(C)(C)C)C1)NCC1(CNC(C2ON=C(CC)C2)=O)CC1 c1(C(N(CCNC(C2CCCC(C)CC2)=O)CC)=O)cc(Cl)c(O)c(Cl)c1 CCCCCCN(C(=O)Cc1cc(C)no1)CCNC(=O)Cn1cc[n+](C)c1 c1(C(=O)NC(C(C)NC(C2(CC#C)CCOCC2)=O)(C)C)ccc2[nH]ccc2c1 c1(C(=O)OC)cc(C)nc(N2CCCC2CN(C)C(c2[nH]c(C)nc2C)=O)n1 C(C(C)(O)C(F)F)NC(C(CNC(COCCC)=O)C)=O C(=O)(CCCCCS(N)(=O)=O)NCCC1CC(NC(c2ccc(C#C)cc2)=O)C1 C1(C)(CC(=O)N(CCC(O)CO)C)CCN(C(c2ccccc2)=O)C1 C1(NC(C=CCCC)=O)C2CC3CN(C(c4nccn5nccc45)=O)C1C3C2 N1(C(C(CC)OC)=O)CCCC(N(C(c2ccc(-c3ccco3)o2)=O)CC)CC1 C1(C(C)(C)NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2cccnc2O)CC1 C(C(CC(=O)NC(CNC(c1ccc(Cl)c(F)c1O)=O)C1CC1)C(F)F)N(C)C c1(C(N2CCC(CN(C(=O)C(C3CCCCC3)F)C)C2)=O)cncc(F)c1Cl c1(CCCC)ccc(C(=O)N(CC(C)NC(=O)C)C)cc1.c1(CN)nc(CC)cs1 N1(C(CC(COC)C)=O)CCC(C)(NC(=O)CC2CCC(=O)C2)CC1 N1(N2C(C(=O)O)CCCC2)CCCC(C(N2C(C=O)CCC2)=O)CC1.C1CC1 c1(CC)ccc(N2CCC(C#N)C2)c2occc12 c1(C(C(C)(C)C)c2ccccc2)nc(C2OCCc3ccccc32)nn1CCF COC1OC(=O)c2c(F)c(C(N3CCCOC(C4CCC4)C3)=O)cc(F)c21 Cc1ccn2ncc(C(N3CC(NC(=O)C(C)(C)CF)CC4(CC4)C3)=O)c2n1 C1(C(NOCCC(C)C)=O)C2CC(O)C(C2)N1C(c1cc2ccccn2n1)=O c1(C(N2C(C)CC(NC(C(C)SC(F)(F)F)=O)C2)=O)ccnc(Cl)c1N N1(C(c2cc(C)oc2C)=O)CCCC(C)(CNC(=O)CCc2cccc(F)c2)C1 C1(NC(c2ccc(C)nn2)=O)CN(C(=O)C(C2CCCCCC2)C)CC1C1CC1 Cc1ccccc1C(=O)NC1CC(O)(CNC(C2(C)CCOC2)=O)C1 c1(C(N2CCN(C(Cn3ncc(C)c3)=O)CC(C)C2)=O)ccc2cccnc2n1 c1(C(=O)NCC(CNC(C(CCC)(C)CC)=O)O)cc2cc(F)cc(F)c2[nH]1 C1(N(C(=O)CCCCC2CC2)CCCN(C2CCCC2)C)CN2CCC1CC2 c1(OC)cccc(CC(=O)NCC(O)CNC(=O)CSCCCC(F)(F)F)c1Cl N1(C(CC(C)OC)=O)CCN(C2CCCN(C(C3CCCC(C)C3)=O)C2)C(=O)C1 C1(NC(C2C(C)(CC)C2)=O)CN(C(c2ccn(CCF)n2)=O)CC1C(F)F C=CC1CN(C(c2cnc(SC)nc2O)=O)CC1NC(c1csc(C)c1C)=O CCCC(C(F)(F)F)NC(=O)C1=CCN(C(C2(OC)CCCOC2)=O)C1 C12CC(C(=O)NCCCN(C)CC)N(C1)C(=O)CNC(=O)O2.C(C)(C)(C)OC.OC C(=O)(CCC(C)(C)C#N)NCCC(C)N(C)C(C1CCCCC1(C)C)=O N1(C(CS(N)(=O)=O)=O)CC2(C1)OC1(CO)CC2(NC(=O)CCN2CCOCC2)C1 c1(C(N2CC(C(C)NC(c3c(C)coc3C3CC3)=O)C2)=O)c(F)ccc(O)c1F c1(C(N(CCCNC(c2cccc(F)c2Cl)=O)C2CC2)=O)ccc2snnc2c1 N1(CC(C2CC2)NC(=O)OC(C)(C)C)CCCC(F)(F)C1c1ccccc1.C(N)(=O)N O(NC(=O)C#CC1CCCC1)CC(=O)NC1CCN(C)C1(C)C C1(NC(c2c(C)scn2)=O)CCN(C(c2[nH]ccc2-c2ccccc2)=O)C(C)C1 C1(C(=O)NC(CC)CNC(c2ccc(C(N)=O)s2)=O)CCCC2(CCC2)O1 C(N=c1[nH]c(C)cc(=NC2CCc3nn[nH]c3C2)[nH]1)C1(C=C)CCC1 CC(C)(CC(F)(F)F)C(=O)NCCC1(O)CCN(C(c2n[nH]c(=N)[nH]2)=O)CC1 c1(C(=O)NCC2(NC(c3csnn3)=O)CCCCC2)ccc2sncc2c1 Cc1cc(C=CC(N2CC(NC(C3(C)CC3(Cl)Cl)=O)CC23CCC3)=O)c[nH]c1=N N1(C(=O)CCF)CCC(NC(C2(C3CC3)CC2)=O)C1 C1(C(N(CCNC(c2cc(C3CC3)[nH]n2)=O)CC)=O)CCN(C(C)C)CC1 CC1(C)C(CNC(c2ccc(C(F)F)o2)=O)CCN1C(C1CCCCC1O)=O Cc1nnc(N2CCC3(NC(=O)CC4CSC4)CCCCCC23)c(C#N)c1C C(=O)(CC(C)(C)C)NCCC(CNC(=O)C(C)n1ccnn1)OC N1(C(c2c(SC)snn2)=O)CCN(C(=O)CN2CC3CC3C2)C2(CC2)C1 CC(C)C(C(=O)NCCCC(C)NC(C1CCCC(=O)C1)=O)NC(N)=O N1(C(C(=C(C)C2CC2)F)=O)CC2(CCCC2N=c2nc3[nH][nH]cc-3c(O)n2)C1 c1(C(=O)NCC2CCCN(C(C3(C#N)CCCO3)=O)C2)nc[nH]c2nccc1-2 Cc1c(C(=O)N(CCCOCCN(C)C(C2C3CCCC23)=O)C)cnn1C c1(C(=O)OC)ccc(NC(=O)C(=O)N(C)CCOCCO)o1 C1(C(=O)NC(C2(O)CN(C(COCCOCC#C)=O)C2)C)CC12CCCCCC2 C1(C(=O)NCCC2N(C(C(CC)CO)=O)CCSC2)CC12CCCCC2 CCCCC(C)(C)NC(=O)C(C1CCCN(C(=O)C(C(C)C)SCC)C1)C N1(C(C(=O)N(C)CC)=O)CCC(C(N2CCC(S)C2)=O)CC1.c1(N)ccccc1Br C(N=c1[nH]cnc2c1SCCC2)C1C(C)CCN(C(c2cnc(NC)cn2)=O)C1 c1(C(N2CC(F)(CNC(c3ccc(F)s3)=O)C2)=O)nn2c(c1Br)CCC2 C1(CC(=O)NCC2CCCCN2CC2CCC(O)C2)CCC=CCC1 C(=O)(N1OC2CCC1C2)C1CN(C(c2cnc(C3CC3)o2)=O)CC12CC2 c1(OC)cccc(C2(C(N3CCC(NC(c4cccnc4O)=O)C3)=O)CC2)n1 C1(NC(c2csc(CNC(C34CSCC3C4)=O)c2)=O)C2COCC12 N1(C(CCSCCC)=O)CC2(C1)CN(C(=O)Cc1csc(C(C)OCC)n1)C2 C1(CNC(C2(C(=O)OC)COC2)=O)(NC(C2(O)COC2)=O)CCOCC1 c1(OC)ncc(C(c2nnnn2Cc2ccco2)NC2C(C)CCC2C)cc1Cl Cc1ccc(C2CC2)cc1NCC1CCC2CC12 c1(SC)nn(C)cc1C(=O)NCC(O)CNC(=O)COc1ccc(C(C)=O)cc1 c1(C(=O)NCC2CC(NC(C(C)C(F)F)=O)C2)cc(F)c(F)cc1N(C)C C1(C(N(C)CC)=O)COC2(CCN(C(=O)CCCNC(C)(C)C)CC2)C1 c1(C(N(C2CCN(C(c3cc(Br)c[nH]3)=O)C2)C)=O)ccc2nc(O)n(C)c2c1 c1(N(CCCCC=C)C)cc(Br)ccc1S(=O)(=O)NC(CCO)C(C)C C1(NC(C2CC(C)(F)C2)=O)CC2CN(C(c3cc4ccccn4n3)=O)CC2C1 Cc1cc(C(=O)N(CCCNC(=O)C(N2CCC(O)CC2)C)C)c(Cl)cc1F Cc1cc(Br)cc(C)c1C(=O)NCc1ccc(CNC(=O)CC(C)C(F)F)cc1 C(C(CO)(CO)NC(C1CC1C1CCCO1)=O)N(C(C(F)=C(C)C)=O)C N1(C(c2c(CC#N)cccc2)=O)CCN(C(C2SC3C=CC2C3)=O)C(CO)C1 C(=O)(CC(C)C(=O)N(CC(C)C(=O)Nc1cn(C)nc1C)C)OC C(CCCCCN(c1ccccc1)C(C1C(C)(C)C1)=O)n1cc(C)nn1.C(=O)O N1(C(C(CC(C)C)(C)C)=O)CCC2CCC(NC(=O)Cc3c(Cl)cnn3C)C1C2 N(C(=NCCc1cncs1)NCC(F)(F)OCC1CCCO1)C(=O)C1CC1 c1(OC)ccc(CN(c2nnc(-c3ccc(C#N)cc3)o2)C)c(Br)n1 c1(C(N(CC(C)NC(c2ccc(Cl)cc2F)=O)C)=O)c(F)cc(F)cc1Cl C1(NC(CCCCSC)=O)CCCC2CN(C(C3Cc4ccccc4C3)=O)CC12 Nc1cc(Cl)cc(F)c1C(=O)NCCC(O)CNC(c1cnccn1)=O C1(CNC(C)=O)CCC2CN(C(c3c(F)cc(F)c(F)c3F)=O)CCC2C1 Cc1ccncc1C(N1CCOC(C(=O)NCc2ccc(Br)nc2)C1)=O C(CC(F)CN=[N+]=[N-])NC(C(CC1CCCC1)NC(c1ccc(CC)o1)=O)=O c1(OC)cnc2c(C)cccn12.C12CCC3CC1CN3CC(=O)N2 C(=O)(CN=c1[nH]c(=NCC2CCSC2)c2ncccc2[nH]1)N(CC)CC c1(N2CCC(C)C(NC(C=CC(CC)=CC)=O)C2C)cc2nnc(C)n2cn1 C1(NC(=O)Nc2scc(C3CN(C(=O)OC(C)(C)C)C3)n2)CCn2cnnc2C1 N#Cc1cc(C(O)C(=O)Nc2ccccc2OCCO)ccc1F c1(C(=O)NC2(COC)CN(C(CC3(COC)CC3)=O)C2)cccc(F)c1N C(=O)(C(C)(F)C(=O)NC1CCN(C(c2cc(C(F)(F)F)cnc2O)=O)C1)OCC C12(NC(=O)OC)CCC(CNC(N3CC=C(CSC)CC3)=O)(CC1)OC2 c1(C(N2CC(c3ccsc3)C(C)C2)C(=O)NC)ccc2c(c1)nc(C)n2C CC1CCCC(C)N(c2nnc(-c3[nH][nH]c(=N)c3Br)n2C)C1 C1(C2CC2)(NCCC(=O)N(C)Cc2ccccc2)CCNC1 c1(OC)cc(NC(C2CC23CN(C(c2ccccc2SC)=O)C3)=O)c(Br)cc1C C1(NC(C2(NC(=O)CC3CCCSC3)C(C)(C)C2)=O)CCC2(CCC2)CC1 N1(C(CC2(C=C)CC2)=O)CCCC(N(C(=O)CCc2cnn(C)n2)C)C1 C#CCC(C)(C(=O)N1CCC(OC(=O)NC)C1)NC(=O)CN(C1CC1)CC C1(C(N(CCC(=O)NC)C)=O)COCCN1C(c1ncccn1)=O C1(NC(C(C(CC)C)C)=O)CS(=O)(=O)N(C)C12CCN(C(C1CC13CC3)=O)CC2 C12(NC(C(OC)OC)=O)CC1CN(C(c1nnn(C)c1C)=O)C2 C12CC(CCC1(F)F)C(=O)OC2=O.C1(N(CC)CC)CCC(C)(C)CC1 C1(C(=O)NCCOCCNC(C=CSC)=O)CCC(F)(F)CC1 N1(C(C2(CCC)CC2)=O)CCC(NC(=O)CSC2CCCCO2)C(O)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CC2CC1(CNC(=O)CCc1cccs1)C2 C(CC(C)N(C)C(c1cnsc1)=O)(C(C)C)NC(CCc1c(C)noc1)=O C1(C(N(c2cc3ccsc3cn2)C)=O)C2CC3CN(C(=O)OC(C)(C)C)C1C3C2 C=C=CCCC(=O)NC1CCCC1CNC(=O)COc1ccc(F)nc1 C1(O)(CNC(C=C(C)Cl)=O)CCN(C(C2CC(n3cc(Br)cn3)C2)=O)CC1 C(CCN=C(NCCC12CCC(CC1)C2)N1CCC(CS(C)(=O)=O)C1)OC CC1CN(C(=O)CCn2cnnn2)C(C)CN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(CC(N2CCC(O)(CNC(CN(C)C3CC3)=O)C2)=O)nc([N+](=O)[O-])n[nH]1 C1(NC(CCCSC)=O)(CNC(c2ccc(C(N)=O)c(Cl)c2)=O)CC2CCC1C2 c1(C(=O)NC2C(NC(c3n(CC)nnc3C)=O)CCCC2)c(N)cc(Cl)cc1Cl Cc1ccccc1N1CCC(NC(=O)NC2COC(CN)C2)CC1 Cc1cc(F)ccc1C1CC1C(=O)NC(C)CC(C)NC(=O)CCCC(C)O C12CN(CCO1)CC(=O)NC2.N1(S(C)(=O)=O)CCC1C(=O)OC C(=O)(NNC(=O)Cn1cnc(C(F)(F)F)n1)C1(C)CCCC1 c1(C(N2CCCCC2CO)=O)ccc(-c2coc3ccccc23)c2cn[nH]c12 C(=O)(C(O)CC(F)(F)F)N1C(CC(=O)NCC(COCC)C)CC2(CC2)C1 CC1OC2(CCN(c3nnc(-c4ccccc4)o3)CC2)NC1=O NC(=O)CCC(=O)NCc1ccsc1C(=O)NCCC(CO)CO c1(C(=O)NC2CCC(CCNC(CC=C=C)=O)C2)ccc(Cl)c(OC)c1N C1(CC(C(=O)NCC2CCOCC2)N(C2CCC(C)(C)C2)C)CCCC(C)(C)C1 Cc1nc2cc(Cl)ccc2n1CC(N1CCNCC1)=O.CC=O c1(C(=O)NC2(C(N3CC(SC)C3)=O)CCC2)[nH]cc2c1CCC2 C1(NC(c2n(C(C)C)ncc2)=O)CC12CCN(C(C1CCCCC1(C)C)=O)CC2 N1(C(CC2CC(=O)OC2)=O)CC=C(CNC(=O)CSc2cn[nH]c2)CC1 N1(C(=O)C=Cc2cnccn2)CCC2CCN(C(=O)CC3CCCS3(=O)=O)C2C1 C(=O)(CC(C)(C)CCC)NC(c1ccccc1F)CNC(C(C=C)C)=O Cc1cc(C(=O)NC(C)CNC(=O)CCCN2CCCC2)ncc1S(N)(=O)=O C(=O)(C(C)C(C)CC)NC1CCC(NC(C(Br)=C(C)C)=O)CC1 CCC1=NOC(C(=O)N(CCC(=O)NCc2ccncc2)CCO)C1 CCS(=O)(=O)CC(=O)N(CC(=O)NCC1(O)CCOC1)C1CC1 c1(C(=O)NC2(C)CN(C(C3C(CC)OCC3)=O)C2)ccc(Cl)c(Cl)c1O C(=O)(C#Cc1ccccc1)NC1CCC(NC(CC(CC)(C)C)=O)CC1 N1(C(c2cc(C(=O)OC)sc2C)=O)CCC(NC(=O)C(OC)OC)C(O)C1 c1(C(=O)NCC2OCCC(NC(c3c(C)ncs3)=O)C2)ncnc2c1CCC2 c1(-c2noc(C3CCCCC3)n2)ccc(N2CCCC(OCCOCC)C2)nc1 C(C)(C)(C(C)CC(=O)NCC(F)Br)NC(c1c(C)nccn1)=O CC1CN(C(=O)CCCCCC#N)CC(C)C1NC(=O)CCCCc1cnc[nH]1 C(=O)(C1=COCC1)NC(CC(C)NC(C(CC)F)=O)C C(=O)(N1C(C)C(=O)c2ccccc21)C1CCCN(C(c2cccc(CC)c2)=O)C1 c1(C(N(CCN(C(CCCOCCC)=O)C)C)=O)ccc(N)c2ncccc12 C1(CCN(C(C(C)OC)=O)CCO)CC2(CO1)CN(C(=O)CN(S(C)(=O)=O)C)C2 N1(C(CSCC(C)=O)=O)CC2ON=C(CNC(c3cc([N+](=O)[O-])n[nH]3)=O)C2C1 C=C(C)CCC(C)NC(=O)C(C1(O)CCC1)NC(=O)Cc1cncs1 C1(NC(c2ccn(-c3ccc(C)cc3)n2)=O)CCC2(CCNC2)CC1 c1(OCC)ncc(C(=O)N(CCCNC(=O)C(O)C2CCCC2)CCO)cc1Cl N1(C(C(CCC)(F)F)=O)CC=C(C(=O)N2CCC2(C)C(C)C)CC1 C(=O)(C1=CC2C=CC(C1)C2)N1CCC(CCC(=O)NC(COC(C)C)(C)C)C1 C(=O)(CC(F)(F)C(F)F)NCCC1(CNC(C2(C(=O)OCC)CCCC2)=O)CC1 c1(C(N2CC3CN(Cc4csc(Cl)n4)CC3C2)=O)ccc2oc(O)nc2c1 C(C1=CCN(C(=O)CC(C)CF)CC1)NC(c1cn(CC(CC)O)nn1)=O c1(OC)ccc(Cl)cc1C(N1CCCC(O)(CCNC(C2(F)CCC2)=O)C1)=O CCC(C)C(C(=O)N(C1CCNCC1)CCN(C)C)OC N1(C(C(C)OCC#C)=O)CC(CNC(=O)COc2ccccc2C)C2(CCC2)C1 N1(C(CCC#N)=O)CCC(CNC(c2cc(-c3ccco3)on2)=O)C(F)(F)CC1 c1(NC(CN(CCCc2c(C(=O)OC)nco2)C)C)ccnc2ncnn12 c1(C(N2CC3C(CNC(C4CC45CCCC5)=O)(C3)C2)=O)cnc2ncccn12 C(=O)(C1=CCCCCC1)NC1C(NC(c2cnc(C(C)C)nc2)=O)C1 C1(NC(C(C(C)NC(c2n[nH]c(C)c2Cl)=O)C)=O)CN(C)CCC1O C(=O)(C(C)(CO)NC(=O)C(C)n1cncn1)NCC(CC)N(C)C N1(C(C2CC3CC2C2CC32)C(=O)NCC=C)CCOCC2(CCOCC2)C1 C1(NC(C(C)O)=O)CCC2CC1CN2C(=O)C#CC1(C)COC1 C=CC(C)(CCOC)C(=O)N1CCOC(C)(CNC(=O)CCc2cnc[nH]2)C1 C(c1cc(C)on1)=C(CC)C.C(C)(C(F)F)=C c1(NC(C)=O)ccc(C(N2CCC(N(C(=O)C(C3CCCCC3)O)CCO)C2)=O)s1 C(F)(C(=O)N(CCC(=O)N1CC(C(=O)OC)C1)CCC)=CCC C1(NC(c2nccc(C)c2)=O)CC(F)CN(C(C2CC(n3cnnc3)C2)=O)C1 Cc1cc(C)c(NC(N2CC(c3nnc(C(C)(C)C)o3)C2)=O)c(Br)n1 N12CC3COCC3(C1)C2=O.c1(OC)ccccc1C(c1ccccc1)NC N1(C(CC)=O)CCC2(CCC(NC(c3sccc3S(C)(=O)=O)=O)C2)CC1 N1(Cc2ccc(C(C)=O)cc2F)CCC2(CO)CCCC12 c1(C(C(=O)NCCCOC)N(C)Cc2ccc(Cl)s2)cccc2nonc12 C1(C(=O)NCC(C(=O)NCCCCC(=O)OC)O)CC2CC1CC2O C1(NC(CCC2CCC(OC)CC2)=O)(CO)CCCN(c2nc(O)nc(O)n2)C1 c1(C(N2CCN(C(CSC)=O)CC2CC(F)(F)F)=O)nc2nc(C)ccn2n1 C(C#Cc1cccc(F)c1F)NC(NC1CC(C)OC(C)C1)=NCC1CC1 CCCCN=C(NCC(C)(C)C(F)(F)F)NCCS(=O)(=O)NC c1(C(N2CC(O)(C(C)NC(C(N3CC(C)C3)C)=O)C2)=O)cccc(F)c1F c1(C(=O)NCc2scc(C(N(C3CC(C#N)C3)CC#C)=O)c2)ccc(CC)cc1 C12(NC(CC=CCC)=O)CCOC(CNC(=O)CCC(C)(C)C)(C1)C2 N1(C(=O)NCC(C)(C)N(C)C)CCC(F)(F)C(C(=O)O)C1 C1(C(=O)NC2C(NC(C3(CC)CCOCC3)=O)C2)CCCCC(C)(C)C1 c1(C(=O)NC2(C)CCN(c3snc(C)n3)C2)ccc(Cl)c(F)c1F N1(C(C(C)OCC)=O)CCCC12CCN(C(=O)Cc1ccc3nonc3c1)C2 c1(CC)cc(NC2CC(NC(=O)CC3CCCOCC3)C2(C)C)nc(C)n1 c1(CNC(c2ccc(Cl)c(Cl)c2)CC)ccc2cc(C)ccc2n1 c1(OCC(C)C)cccc(CNC(c2nnnn2C)(C)Cc2ccc(Cl)nc2)c1 Cc1cc(C)c(C(=O)NCC2CC3(CC(NC(=O)Cc4cc[nH]c4)C3)C2)c(O)n1 c1(CC(=O)OCC)n[nH]c(=NC2=NCC(n3cc(P(C)(C)=O)cn3)C2)s1 C#CCC(C)(C)C(=O)NCC1CC2(CC2)CN1C(=O)Cc1n[nH]c(=NC)s1 c1(C(C(N2CCN(C(c3cccc(COC)c3)=O)CC2)=O)C)cccc(C#N)c1 c1(C(=O)N(CCCNC(C2CC3CCC(C2)O3)=O)C2CC2)cc2ncccc2s1 C=C(CN(C(C1CC(OC)C1)=O)C1CC1)CCNC(=O)C(c1cnccn1)C c1(C(=O)Nc2nc3cnccc3s2)cc2cn[nH]c2cn1 Cc1ccc2ccn(CC(=O)NC3CCC(NC(=O)C(C)(O)C4CCC4)C3)c2c1 N1(C(C2(CC)CCC2)=O)CC2C(CNC(=O)Cc3cccc(O)c3)C2C1 C1(CN(C(C2CCN(C(C)=O)C2)=O)C)CCN(C(=O)CC2CCCC(C)C2)CC1 c1(CC)nnc(C)cc1C(N1CCC(CNC(=O)CC2CC2)(OC)CC1)=O c1(OCCC)nc(C)ccc1C(=O)N(C)CCNC(C1(c2ccnn2C)CC1)=O c1(C(=O)NCCN(C(c2ccc(C(C)C)s2)=O)CC)cnc2[nH]c(C)nc2c1 Cn1cccc1C=CC(N1CCCC(C(N2CCCC2)=O)C1)=O N1(C(c2c(C)cncc2)=O)CCCCC12CC(NC(=O)CCc1cnn[nH]1)C2 C(=O)(C(CC(F)F)NC(c1c[nH]nc1[N+](=O)[O-])=O)NCCCCS(C)=O c1(C(N2C(C(C)NC(C(=O)NCCOC)=O)CCC2)=O)cc(OC)ccc1OC C1(NC(CCOCCC)=O)CCN(C(=O)CCc2cnn(C)n2)C1(C)C N1(C(COCC(C)C)=O)CCCOC(C(=O)NC2CC2CCN(C)C)C1 CC1CCN(CC(N2CCC(C(N3CCCC3CN(C)C)=O)C2)=O)C1 C1(C(N2CC(C#C)C2)=O)CNC(=O)CN1C(c1ccncc1)=O [N-]=[N+]=NC1CN(C(C2OCCC2NC(C2CCC3CC2CO3)=O)=O)CC1O c1(C(N(C)CC2CN(C(C(C)c3ccsn3)=O)C2)=O)ccc(-c2ccccn2)s1 C1(NC(c2csc(CO)n2)=O)CC2(CCN(C(=O)C(F)CC3CCCC3)CC2)C1 C1(CC)C(NC(c2ccncn2)=O)CCCN1C(C1CC(C)=NO1)=O C(C1CSc2ccccc21)NC(c1ccnn1C1CCNCC1)=O C1(C(=O)NCCCN(C(C2(CC(C)C)CC2)=O)CCO)CCOCC1C(C)C c1(NCC(F)(F)Cn2cc(CO)nn2)ncnc(C)c1Br.c1(NCC)ccccc1O c1(C(N(C2CCCN(C(C(C)OC)=O)C2)CCF)=O)nccc2occc12 c1(NCC2N(C(C3(F)CCS(=O)(=O)C3)=O)CCC2)nc(O)c2c[nH]nc2n1 CC1(C)COC(CC(N2CCC(CNC(=O)CCCC3CC3)C2)=O)CO1 CC(C)N=C(NC1CCC1)NCC(c1cc(F)cc(F)c1)O C(CCN=C(NCC(C)C)NCc1ccc(CC2(Br)CCC2)cc1)SC C1(CNC(CC(C=C)C)=O)CC(O)C(O)CC1C(=O)N(C)Cc1cnn(C)c1 C1(NC(CNC(=O)OC)=O)CC12CC(NC(c1ccn(C3CCCC3)n1)=O)C2 n1(CC(=O)NC2CN(C(c3cnn[nH]3)=O)CC3(CC3)C2)cc([N+](=O)[O-])ccc1=O C1(NC(c2c(CNC(CCOCCOC)=O)c[nH]n2)=O)CCCCC1(F)F C1(NC(C2CCC2C(=O)NC)=O)CCOC(CNC)C1.C1(CC(=O)OC)(COC)CC1 C=C(Cl)C(C)(C)C(=O)N(CCCN(C(=O)CC1CC(O)C1(C)C)C)C C(=O)(C(C)(F)C(=O)NCc1nc(CNC(c2cnc(O)s2)=O)cs1)OC c1(C(N2CCCN(C(CC3CC(=C)C3)=O)CC2C)=O)cc(C)nc2c1cnn2C c1(C(N2CCCN(C(C3CC(=C)C3)=O)CC2CO)=O)cc2ncc(CC)cc2[nH]1 N1(C(Cc2ccc(OCC)cn2)=O)CCN(C(c2scnc2C)=O)C(C)C1 CC(c1ccsc1)=CC(=O)NCC(C)CN(C(=O)C(CO)N(C)C)C c1(NC(C2CCC(NCc3ccc(OC)nc3)C2)=O)cc(C)cc(Cl)c1 C(=O)(C1CCCn2ncnc21)NC(CN(C(C=Cc1cncc(OC)c1)=O)C)C C(=O)(CCCC(=C)C)N1C(CNC(=O)COCCC(F)(F)F)CC(OC)C1 C1(C)(C(N2CCCC(N(C(CN(C)CC)=O)CCO)C2)=O)CC(C2CC2)=NO1 c1(SC)cc(CC(=O)NCCC2(CNC(=O)C(CC)OC)CCC2)ccc1OC c1(N(CCCCN(C)C(c2conc2-c2ccccc2)=O)C)ncnc(=N)[nH]1 c1(C(=O)NCC2CCCN(Cc3cn(CCF)nn3)C2)ccc2ccoc2c1 C(=O)(C1=NNC(=O)CC1)N1CCC(N2CCN(C(C3C(C)CCO3)=O)CC2)CC1 N1(C(C2(CC=C)CCOC2)=O)CC=C(C(=O)NCC(c2ccccc2)O)CC1 C1(C2CCCO2)(C(N(CCN(C(=O)Cc2cnn(C)c2)C(C)C)C)=O)CCCC1 Cc1c(NC(C2CCN(C(=O)CC3CC3)C2)=O)ccc(Br)c1Cl c1(CC)cc(C(=O)NCC=CCNC(c2ccc(C(C)F)cc2)=O)cc(Cl)c1 c1(C(=O)NCC(CC)NC(=O)C(c2cnccn2)C)n[nH]c(C)c1Cl C1(C(N(CCC)CCNC(c2nnsc2SC)=O)=O)CC2C(C1)C2(F)F n1(CC#C)c(C)cc(C(=O)NC2CCC(NC(=O)CC(O)C(C)C)CC2)c1C c1(N2CC2c2ccccc2)ccc2ccccc2c1[N+](=O)[O-].C1(C(C)O)CCCC1 n1(CC(=O)NCC#CCNC(=O)C(F)C(F)(F)F)ncc2ncccc12 C(=O)(C1=CCCC1C)NCCC(C)N(C)C(c1coc(CC2CC2)n1)=O c1(C(=O)NC(C2CCN(C(CSCCCC)=O)CC2)(C)C)cc(C#N)n(C)n1 c1(CNC(COCCOCC)=O)cc(C(F)(F)F)c(O)c(N)c1.C12CN(C1)C2=O c1(C(=O)OCc2cccc(Cl)c2)c(F)cc(N(C(C)(C)C)C2CC2)c(F)c1F n1(CC(N2CCN(C(=O)CNc3ncccn3)C(CF)C2)=O)cc([N+](=O)[O-])cn1 N=c1nnn(CC(=O)NCCNC(C2C(CNC(c3ccoc3)=O)C2)=O)[nH]1 CC(C)(Cc1ccccc1)CC(=O)NCC1COC(CNC(=O)Cc2ccoc2)C1 N1(C(C(CC)n2cncn2)=O)CCCC(NC(c2c[nH]cc2C2CC2)=O)C1 CC1=CCC(C(=O)NC(CN(C)C)C(=O)NCC(=O)NC(C)(C)C)CC1 C1(CC(=O)NCC(C(C)C)(C)NC(c2cncc(F)c2)=O)CCCCC(=O)N1 c1(C(N2C(C(=O)NC(C)Cn3ccnc3)CC3CC32)=O)nccc2cc[nH]c12 C1(CNC(=O)C(O)C2(O)CCC2)CCCCC1O CC(C)C(C(=O)NC(C1CCN(C(=O)C2=NOCC2)CC1)C)N(S(C)(=O)=O)C1CC1 C1(NC(C2(CF)CCN(C(CCCOC)=O)C2)=O)CN(C)C2(CCC2)C1 CC(CN=c1c(C#N)c[nH]c2c(F)ccc(Cl)c12)N(C)CC1CCC1(C)C c1(OCC(=O)NCC(CN(C)C)O)cc(C(F)(F)F)cc(Br)c1 C1(C(N2CC(NC(C(C)(C(C)C)OC)=O)C(C)C2)=O)CC2(C1)CC(F)(F)C2 c1(N(C)Cc2ccc(OC)nc2)nc(N2CCC(F)C2)nc2cccc(F)c12 Cc1ccc(O)c(NC(C2CC(C)CN2C(c2cc(Br)cnc2O)=O)=O)c1 N1(C(C)=O)CCC(C(=O)Nc2cccc(NC(C3(N(C)C)CCC3)=O)c2)CC1 C1(CC(=O)N(CCSC)C)CC2(CCCC2)CO1.C1CCO1.C(=O)N.C1COCC1 C1(OC)(OC)CC(C)(C(C)NC(=O)CC2CCOC2)C1.C(C)(C)(C)OC(=O)C1CC1 CCC(CC(F)F)C(=O)N1CCC(N2CCN(C(=O)CC(C)CC(C)C)CC2)C1 C1(C(=O)NCC2(F)CCN(C(c3cc(F)c[nH]3)=O)C2)Cc2cccc(F)c2O1 N1(C(CN(C(CSCCC(C)C)=O)C2CCC2)=O)CCC2CC2C1 c1(C(=O)NC2CC3CCC2N3C(C23CCC(CC2)C3)=O)cc(Cl)c(F)cc1F C(Cc1c(F)cccc1F)(C(=O)N(O)Cc1cn(CC)nn1)n1c(SCC)nnc1 C12(C(N3CCC(C(CNC(Cc4ncc(C)[nH]4)=O)C)CC3)=O)CCC(CC1)CC2 C1(F)(CNC(Cc2[nH]n(C(C)(C)C)c(=O)c2)=O)COCCN(C(C23CC2C3)=O)C1 Cc1cnc(C(N2CCCC2C2(NC(C3CN(C)CCO3)=O)CC2)=O)cc1C N1(C(C2(C)CC2)=O)CC2(CC2C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 c1(C(=O)NCC=CCNC(=O)C=C2CCC2)cc2ccc(Br)cc2o1 c1(OCCC)ccc(C(=O)NC2COCC2NC(=O)C(F)OC)cc1 c1(OC(C)=O)cccc(C(N2CSCC2C(N2CC(C)(O)C2)=O)=O)c1C CCC(CC)CC(F)C(=O)NCC1CC12CCN(C(=O)C1=CC(C)C1)CC2 c1(NC(C2CN(Cc3cc(O)ncc3Br)C2)=O)c(F)cc(C(F)(F)F)cc1F Cc1coc(C(=O)NCC(O)CNC(=O)Cc2cc(C(F)(F)F)nn2C)c1C c1(C(=O)NCCN(C(C2C(CC)CCC2)=O)Cc2ccccc2)cn(C)cc1C C1(NC(C(=O)NCCCC(N)=O)=O)CC1C1CCOC1 c1(C(=O)NCC2(NC(C3C(=C)C3)=O)CCOC2)cnn(CCC(C)C)c1C c1(CC)nc(CC)ccc1C(=O)NCC(CO)NC(=O)CC1CCCC(C)(C)C1 Cc1cc(C(N2CCC2(C)CC(=O)NCC2CCCCN2C)=O)cc(C)c1 Cn1[nH]c(=NC(=O)NC2(c3cc(F)cc(C#N)c3)CC2)cc1OC N1(C(c2c(C)sc(O)n2)=O)CCCC(C)(CNC(c2cnn(C(C)C)c2C)=O)C1 Cc1cccnc1CCC(=O)NCC(C1CC1)NC(c1ccc[nH]1)=O Cc1cc(C(=O)N(C)CC2CCN(C(C3CCCOC3)=O)C2)[nH]c1C CC(=O)CC(C)(C)C(=O)N1CCC(C(=O)NCC2CC3C=CC2C3)(CF)C1 C(c1cccc(C2CCN(C(C3CN(C)CCO3)=O)CC2)c1)=CCCC Cn1ncc([N+](=O)[O-])c1NC(=O)Cc1ccccc1NCc1cccc(O)c1F C(N=c1[nH]c(=NCCOCC2CCC2)[nH]c2c1CCCC2)C1N(C)CC(O)C1 CC1CN(C(c2ccc(CO)cn2)=O)CC(C)N(C(=O)CO)C1 c1(NC(C)=O)cc(F)c(F)cc1C(=O)NC1CCN(C(c2cncnc2C)=O)C1 C1(CCNC(=O)NCC(=C)C(F)(F)F)CC(C)OC(C)C1 C1(NC(c2c(C)onc2)=O)CN(C(C2CCCCNC2=O)=O)CC2(CC2)C1 N1(C(C2(C#N)C(C)C2)=O)CCC2(CCCN2C(c2cc(C(F)F)ccn2)=O)CC1 N12CC3(CCC1CC3)C2=O.C1(C2(NC(C3(CSC)CC3)=O)CC2)CCCCO1 c1(NC(C2CC3CC3N2CC2(c3ccccc3)CC2)=O)ccc(C2CCOCC2)cc1 C1(C(=O)Nc2c(I)ccc(C#N)c2)CCCC12CCN(S(=O)(=O)C(F)(F)F)C2 C(C(O)CNC(C1CCOC1)=O)N(C)C(C1CC(CC(C)(C)C)C1)=O C1(C(=O)OCc2ccc(CC(=O)OCC)cc2)(CC)CC2(CCC2)C1 c12cc(cc(Br)c1)C(NCC1CCCN1S(C)(=O)=O)CO2.CCCCC c1(C(N(C(C)CNC(=O)C2=CCCC2)C)=O)ccc2cccc(O)c2c1 N1(C(CCC#N)=O)CCC2(NC(=O)CCc3c(F)cccc3F)CCCCCC12 N1(C(=O)Cc2ccoc2)CCC2(C1)CN(C(C1CC3CCC1C3)=O)CCO2 N1(C(Cc2ccn(CC)n2)=O)CCCC(C)(C)C1CC(=O)NC1CCCN(C)C1 C1(NC(C2C(CNC(CC(C)=C(C)C)=O)CCO2)=O)CC12CC(O)C2 C1(CNC(C(=C(C)C2CC2)F)=O)(NC(=O)CNc2nccs2)CC2CCC1C2 C1(COC)(CSC2CC(OC)CN2C)CCN(C(=O)OC(C)(C)C)C1 C(C(=O)NCCn1ncc(C)c1)(C(C)CC1CC1)N(C(C)(C)C)C CC1=C(C(=O)N2CC(CNC(C3(CF)CC(c4ccccc4)C3)=O)C2)CCCC1 C1(CC(C)NN2CCCCC2)N(C(N)=O)CC1(C)C.n12cc(nn1)CN1CC2C1 N1(C(CC=C)=O)CCC(C2CCN(C(c3cc(CC)ccc3OC)=O)CC2)CC1 c1(C2CN(C(=O)N(C3(CO)CCNCC3)C3CCCOC3)C2)ccc(F)c(F)c1 n1(CCC)nccc1C(N1CCC1C(=O)NCc1sccc1CC)=O C12CC13CCN(C3)C2=O.c1(NC(C(C(F)(F)F)NC(=O)C2CC2)=O)cccc(Cl)c1 c1(C(=O)NCCN(C)C(C2CCCC(N(C)C)C2)=O)cnc2c(Cl)cccn12 c1(C(C)NC(c2cccc(Cl)c2)C(C)C)cccc(Br)c1Cl N1(C(c2nn(C)c(C(F)(F)F)c2Br)=O)CC(N)CC2(CCC2)C1 C1(CNC(CS(=O)(=O)NC)=O)CC2(CCC2)CN1C(c1c(Cl)nsc1Cl)=O N(C(=NCCc1cccc(C)n1)Nc1ccc(OCC)c(OC)c1)CCOC C(=O)(CC(CC)C(C)C)NCCOCCCNC(C1N(C(C)=O)CSC1)=O C1(NC(=O)NCC(COC)O)CCCC(C2CC2)C1 N1(C(CSC)=O)CCOCC1C(=O)Nc1ccc(-c2ccccc2)nc1 c1(CN2CC(NC(c3c(OC)cc(I)cc3)=O)C(F)C2)cc(C)cc(Br)c1O CCN(OC)C(=O)CCC1COCCN1C(c1cc(C2CC2)on1)=O N1(C(CC2N(C(C(C)=C3CCC3)=O)C3C2CCC3)=O)CC2CCC(C1)C(=O)N2 C1(C(N(C(C)C(=O)N(CCC(N)=O)C2CC2)CC)=O)C2COCC12 c1(C(N2C(C(=O)NCc3c(C)cncc3)CCC2)=O)cc(Br)cnc1O Cc1cc(C(N)=O)cc(CNC2CC2C(N2CCS(=O)(=O)CC2)=O)c1 N1(C(C)(C)C)CC(C(=O)NC2CC(CCNC(c3cnn(C)c3F)=O)C2)CC1=O c1(OC)ccc(CN2CC3C(C(=O)NC(CO)C4CC4)C3C2)c(OC)c1 C1(NC(c2cn(C)nc2Cl)=O)CC2CC1CN(C(c1cc(Cl)c(F)cc1F)=O)C2 Cc1cc(C)c(CC2OCCN2C(=O)Cc2cccc(F)c2F)c(C)c1 C(CCN=C(NCCn1c(C2CC2)nc2ccccc12)N1CCC(C)(F)C1)OC C1(c2nnnn2Cc2ccccc2)(NC(CCCC)(C)C)CC2(CCC2)C1 C#Cc1ccc(C(N2CC3(CC(NC(C4CN(C5CCOC5)C4)=O)C3)C2)=O)cc1 c1(OCC)cccc(CN2CCC(CCNC(=O)CCc3ccncn3)CC2)c1 c1(COC)cccc(C(=O)NCC2CCCC2C(=O)N(C)CC2CCCN2C)c1 N1(C(C2C(CC)CCO2)=O)CC2CC2(CNC(c2nn(C)cc2C)=O)C1 C1(C(N2C(C)CCCC2C)=O)COC2(CCN(C(=O)C(c3ccccc3)F)C2)C1 c1(OC)ccc(F)cc1C(=O)NCC(C1CCCC1)NC(=O)C1=CCCO1 N1(C(c2c(C)onc2O)=O)CCN(C(=O)C(C)Oc2ccccc2Cl)C2(CC2)C1 CC(C)CC(CNC(=O)CN1CC2CC2C1)C(=O)NCC1CCN(C2CC2)C1 CS(C)(=O)=NCC(=O)N1CCCCC1C1CCN(C(c2ccc(F)cc2Cl)=O)C1 CCS(=O)(=O)N(CC(=O)NCCCN(C(=O)CN(C1CCCC1)C)C)C n1(CC)cnc2ccccc12.N12CCC(C(C)C1)Nc1c2nccc1.CO c1(CC(=O)N(C)CC2OCCN(C(C(C(C)C)(C)O)=O)C2)ccc(S(C)=O)cc1 Cc1c(C(=O)NCC(O)CNC(c2cn(C)c(=O)n2C)=O)[nH]c2c(C)cccc12 CCCC(C)CC(=O)N1CC(F)(CNC(=O)CC(C(F)F)N2CCOCC2)C1 N1(C(C(n2c(C)ncc2)C)=O)CCC(C)(CNC(=O)C(c2cccnc2)C)CC1 C1(NC(c2ccsc2)=O)CCCCC12CCCN(C(c1cc(Cl)nc(Cl)c1)=O)C2 N1(C(C(c2ccc(C)s2)C)=O)CC(NC(C2(F)CCOCC2)=O)C(O)C1 C(C)(C)(CCCC(=O)NCC1CCC1)NC(C(CC=CC)C)=O c1(C(=O)NCC(c2ccc(F)c(Cl)c2)C)cnn2cc[nH]c12 C12CCCCCCC1n1cc(nn1)C1(CC1)C(=O)N2.N1(CO)CCC(=O)NC1=O C1(CNC(COCCOC)=O)CC2(CCC2)CN1C(=O)CC1CCCCO1 Cc1n[nH]c(=NC2C3CC2CN(C(=O)CCCCC2CCCCC2)C3)o1 N1(C(CN2C(NC(c3nc(NC(C)=O)sc3)=O)CC2)=O)CCSCC1CCOC c1(C(=O)NC2C(NC(CCCCSC)=O)CCC2)sc2cccc(F)c2c1Cl N1(C(C(CC#C)O)=O)CC(C)(C)CC1CNC(c1[nH]cnc1CC)=O N1(C(CC(CNC(C(CCCOC)C)=O)(C)C)=O)CCOC2(CCC2)C1 c1(NC(C2(C)CCCN(C(CC(=O)OC)=O)C2)=O)cc(OC)c(OC)cc1C C1(C(N2C3CC(NC(C(N)=O)=O)CC2CC3)=O)CC(c2ccc(F)cc2)=NO1 Cc1cc(C(=O)NCC(CC(C)C)NC(C2CC(C)N(C)C2)=O)ncc1C(F)F c1(CC(N2CCN(C(C3CCC3)=O)CC(O)C2)=O)coc2c(Cl)c(Cl)ccc12 C(=O)(C1Cc2ccc(F)cc21)NC1C(NC(CCOCC#C)=O)CS(=O)(=O)C1 N1(SCC)CCC(N2CCC(NC(=O)Cc3cc(=O)n(CC(C)C)[nH]3)CC2)C1=O c1(OC)ccc(C(=O)N(CCNC(C2(C)CC3(CC3)C2)=O)CSC)cc1OC CC1(c2cn(Cc3csc(Br)n3)nn2)CCN(C(C2(S(N)(=O)=O)CCC2)=O)CC1 C1(C(=O)NCCN(C2CCCC2)C)CN(C(c2ncccn2)=O)CC1(C)C C=CC(C)(C)C(=O)NC(C)CC(C)NC(=O)Cc1cc(C2CC2)nn1C Cn1cc(N=c2[nH][nH]c(=NC(CF)c3ccccc3F)cc2Cl)cn1 C=C1CCC(CNC(=O)C(CCC)NC(c2ncccc2O)=O)CC1 C1(CNC(COCCCC#C)=O)CCCCN(C(c2ccc(CO)nc2)=O)C1 N1(C(C(C)OCCN(C)C)=O)CCC(F)(CNC(c2csc(Cl)c2)=O)CC1 c1(OC)cc(C(=O)NC(C2CCN(C(=O)CC3CCC(C)CC3)C2)C)ncn1 C1(C(N(CCNC(=O)CCc2nnc(C3CCCC3)o2)CC)=O)CCS1(=O)=O CCCCCCN(C)C(=O)NCC1CC1CNC(=O)OC(C)(C)C N1(C(CSCCCC)=O)CC2(CNC(=O)C(CC(C)C)N(C)C)CC1CCO2 CC1C(=O)CC2CCC1N2C(=O)Nc1ccc2c(c1)CCN2 C1(NC(C2CC(NC(C3N(C)CCCCC3)=O)C2)=O)CCCOC12CCC2 c1(CNC(CNS(CCCOCC)(=O)=O)=O)c(Cl)ccnc1Cl N1(C(Cn2ncc(CC)c2)=O)C2CCC1C(CNC(C1CC1(C)C)=O)C2 C(=O)(C(O)CC(C)C)NCC1(C(N2C(C(=O)OC)CC2)=O)CC=CC1 C(=O)(C(CP(C)(C)=O)P(C)(C)=O)NC12CN(C(C3CC(SC)C3)=O)C(C1)C2 c1(C(=O)NCCN(C(C)C)C(c2cnc(Cl)s2)=O)ccc2c(c1)C(=O)NC2=O C1(NC(=O)CCc2nccs2)CC2CCC1N(C(=O)CC1CCCC1)C2 c1(N(C)C)ccc(N(CC(c2ccccc2)OCC(=O)N(C)C)C)cc1 c1(NC(=O)NCC2CN3CCC2CC3)cc(Cl)cc(Cl)c1F c1(Cn2cc(CC3N(C(CC(=C=C)C)=O)CCC3)nn2)ccc(F)cc1F C1(CCNC(C2(CC)CC2(F)F)=O)CN(C(C2(F)CCCCC2)=O)CC(C)O1 N1(C(C)=O)CCOCC1C(=O)NC1CCC(CNC(=O)CCCn2ccnn2)C1 c1(OC)ccccc1C(N1CCC(F)(C(=O)NCCCP(C)(C)=O)C1)=O c1(C(=O)NCCN(CCC)C(c2cnc(C3CC3)o2)=O)cc(Cl)cc(Cl)c1 CC1(C)C2CC1CN(C(C1CSCCN1C(=O)CC(F)(F)F)=O)C2 C1(OC)CN(C(C2CCCO2)=O)CC1C(N1CCCC1CC1CCCC1)=O N1(C(c2ccc(SC)o2)=O)CCC2CC12C(=O)NCCCC1CCOC1=O c1(C(N2CCC(C(F)F)CC2)C(=O)NCCC)ccc(C(=O)OC)cc1Br CC1(C)OCCN(C(=O)C(Cc2cccc(Br)c2)C(N)=O)C1CO C=CCC(C)(CC)C(=O)NCC1CC2(C1)CN(C(C1(C)CC3CCC1O3)=O)C2 C12(C(=O)NC(COc3cccc(C)c3)C)CC(CN)(C1)OC21CNC1 C1(C(=O)NCC=C2CCN(C(C(CC(=C)C)C)=O)CC2)CC2OC(=O)OC2C1 N1(C(c2nnn(C)n2)C(=O)NC2CC(F)(F)C2)CCN(Cc2nc[nH]n2)CC1 c1(N2CCC(C)(Nc3nccc(N4CC(C)OCC4)c3)C2)ccc(F)cc1F c1(OC)cc(C(=O)CCC(=O)NCCNC(=O)CSC(F)F)ccc1F c1(C(=O)NCC2N(C(C(C(C)O)C)=O)CCCC2(C)C)ccc2nccnc2c1 Cc1cc(=NCC2OCCOC2(C)C)[nH]c(=NCC(C)(C)CC(F)(F)F)[nH]1 C=C(Cl)CC(C(=O)NC(CCCC)C(=O)NC)NC(C1CCCC1C(C)C)=O C1(C(=O)NC2CC3(C(NC(c4cnc(OC)s4)=O)C3)C2)CC12CCS(=O)(=O)CC2 C1(CNC(c2cc(C(C)C)[nH]n2)=O)CN(C(C2CC3(CC(=O)N3)C2)=O)C(C)(C)C1 c1(C(=O)NC2C=CCN(C(=O)C(O)C3CCCC3)C2)cncc2nc[nH]c12 c1(C(N2CCC3C(NC(c4ccc(OC)cc4)=O)C32)=O)nccc2[nH]ccc12 C=CC1(CC(=O)NC2(CN(C)C)CC2)CN(C(C2CCC(CC)CC2)=O)C1 C1(C(=O)NCCCCC(C)NC(C(CCSC)(C)C)=O)CCC2C(C1)C2(F)F c1(C(=O)NCC(N2CCC(C)CC2)=O)cc2c(Br)csc2[nH]1 N1(CCC)CCC(NC(C2CC(NC(c3nocc3Cl)=O)CCO2)=O)CC1 N1(C(COc2snc(C)n2)=O)CC(F)(F)CC1Cn1cc(CCCC#N)nn1 c1(C(C)C)nc(NCC(C)CCO)cc(N2CCC(CCCO)C2)n1 C(=O)(C1OCCc2cc(O)ccc21)NCCC(N1C(C)C(C)SCC1)=O N1(C(C(CC)(C)CO)=O)CCN(C(C2OCCCC2(C)C)=O)C2(CCC2)C1 Cc1n[nH]c(C)c1CC(C)C(=O)NCCNC(C1CCCCN1c1ncccn1)=O c1(OC)ccc(C(N2CCCC2CCC(N2CC=CCC2)=O)=O)cc1F C(=O)(C(C)C(=O)N1C(C(=O)NCCC(C)F)CCC1C(C)C)OC C1(NC(Cc2c(C)ocn2)=O)CCN(C(=O)CC23COC(C)(C2)C3)CC1 CC1CCN(C(C2C(C)(C)C2(C)C)=O)C(CNC(=O)Cc2ccsc2Cl)C1 N1(C(C2C(C(=O)OC)C2)=O)CCC2(CCN(C(C3C4CC(=O)CC34)=O)CC2)C1 C(=O)(CCCCCC#N)N1CC(CC(=O)NCC(C)C(C)(C)C)OCC1 N1(C(C(C)(C)N2CCCC2)=O)CCOCC(F)(CNC(C2(C(N)=O)CC2)=O)C1 C1(COC)CN(C(C2CC(=O)N(C)C2)=O)CCN1C(c1ccccc1C(N)=O)=O C1(C(=O)N(CC(C)(C)NC(=O)C(C)NC(N)=O)C)(COC)CCOC1 c1(OC)coc(C(=O)NC(C)CN(C(=O)CCOc2ccc(Cl)cc2)C)cc1=O CCC(C)(CCNC(c1cc(C)nn1CC)=O)NC(c1cncc(F)c1)=O C=CCCCCCCCC(=O)NCC1CC1CNC(=O)CCc1cncnc1 N1(C(c2c(C)snc2)=O)CCC2(CCN(C(C3(CS(C)(=O)=O)COC3)=O)C2)C1 N#CC1(NC(C2CCN(C(c3c(I)ccnc3Cl)=O)CC2O)=O)CCOCC1 C(CC1=CCOCC1)NC(C1C(NC(C(C(=O)OCC)F)=O)C1(C)C)=O C1(C(=O)OC)C2CC3C(C2NC(C24CCC(CC2F)C4)=O)C13 N#Cc1cccc(CCC(=O)NC(CNC(=O)Cc2cnn(C(F)F)c2)C2CC2)c1 C1(CNC(CCN(CCC)C)=O)CC(F)CN1C(C1CCC(C)(CC)O1)=O N1(C(c2c(C)cc(C)o2)=O)CCCC2CN(C(C3CCC3C(C)(C)C)=O)CCC12 C1(NC(C2(F)C(C)C2)=O)CC2CCC1CN(C(c1onc3ccccc13)=O)C2 Cc1c(NC(C2CC(C)CN2C(=O)C(=O)N(C)C)=O)cccc1CO C1(C(=O)NCC(=O)NCC(c2ccccn2)C)CC2(CCCCC2)S1(=O)=O C1(NC(=O)CCC2OCCO2)CC2CCC1C(NC(c1cnc(C(F)F)s1)=O)C2 N1(c2ccc(OC)c(OC)c2)C(=S)NC(c2ccc(I)s2)C2=C1CCCNC2=O C1(C#N)(C(=O)NC(CC#C)C(=O)NC2CC(C)(CC)C2)CCCOC1 C1(C(N2C(CN(C(c3cc(C)ccc3F)=O)CC)CCC2)=O)C2(CCC2)C12CCC2 Cc1cc(C(=O)NC(C)(C)CNC(=O)C(F)=CC2CC2)cc(C)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(c2c[nH]nc2C)=O)CC(O)C1 C(=O)(C(C)(C)CC(=O)N1CC(OCCNC(c2nc(Br)c(C)s2)=O)C1)OC CC1CC(C)(C(N2CC(NC(C3CC(N4CCN(C)CC4)C3)=O)C(O)C2)=O)CCO1 N1(C2CCN(C(c3cc(C(C)=O)sc3)=O)C2)CC(NC(c2cocn2)=O)CC1=O N1(C(=O)CCOC2CCOC2)CCC2(CC1)CN(C(C1CCC1(F)F)=O)C2 N1(C(C=CC(CC)=CC)=O)CC2CC1CC2NC(=O)C=Cc1ccc(CC)o1 C1(NC(=O)CN2CC3CC3C2)CCN(C(c2ccc(C3CC3)cn2)=O)CC1F C(CCC(C)C)(C(=O)NCC1(CC(C)C)CC1)NC(C(C(=O)OC)OC)=O CC1COCCC1NC(C1(NC(C2CC3(CCC3)C2)=O)CCCCC1)=O C1(C(N2C(CNC(c3ccc(OC)nc3C)=O)CCC2)=O)CCCC2(CCC2)C1 C(=O)(C(O)C1CCc2ccccc21)N1CCCCC(CNC)C1 Cc1cc(=NC(C)CN(C(=O)CC(C)C(C)C)C)[nH]c(S(C)(=O)=O)n1 C(=O)(C1CCc2cccnc21)NC(CNC(c1c(Br)cc(C)s1)=O)C C12(NC(=O)COCC3CCCC3)CCCN(C(c3cccc(Cl)c3)=O)CC1C2 CCC(C(=O)NCCOCCN(C)C(c1sncc1C)=O)C1CCC(=O)N1 C#Cc1ccc(OC)c(C(=O)NCC=CCNC(=O)CC2OCCC2C)c1 N1(C(CS(=O)(=O)NC)=O)C2CCC1C(NC(C1(C)CCC13CCC3)=O)C2 Cn1cnc2nc(=NC(C)(C)CCNCC(c3cccnc3)(C)C)[nH]c(C(N)=O)c12 c1(C(=O)OC(C)(C)C)ccc(N2CCOC(CCC(F)(F)F)C2)nc1 C(=O)(CCCCCF)N(CC)Cc1cn(CCNC(C2CC3C=CC2C3)=O)nn1 CC1CSCCN(CC(=O)N(C)C(c2n[nH]cn2)c2ccco2)C1 N1(C(C2(C)CCN(C)CC2)=O)CCC(N=[N+]=[N-])(C(N2CCC23CCCC3)=O)C1 N#Cc1c[nH]cnc1=NCC1CCC2(CCC2)C1NC(c1cncnc1)=O C(=O)(C(O)C(F)(F)F)NC1CC(CCOC)C1.c12cccc(c1)NC2=O N(C1CCCc2sc(Cl)cc21)Cc1oc(C)c(C)c1C(=O)O N1(C(c2ccc(C)cc2O)=O)CCC(C)N(C(=O)CC2CC(O)C23CCC3)CC1 n1(CCC)cc(CNC(C2CCC(Nc3ncc(C(F)(F)F)s3)C2)=O)cn1 C1(C(N2C(C(=O)OC)C(C)(C)C2)=O)CCCC2(C1)OCCO2 c1(OCC(=O)NCc2scc(CNC(c3c(C)ocn3)=O)n2)ccc(Cl)cc1F C(CCC(C)CC(=O)N1C2CCC1C(NC(=O)CCC(N)=O)C2)=C(C)C C1(SCC)CCC(C(N2CCOCC2CN(C)C(C2CC2(C)C(F)F)=O)=O)CC1 c1(NC(CCC2CC(NC(CCCOC)=O)C2)=O)cc(C)ccc1Cl N(C(=NCC1CC=CC1)NCc1nsc(-c2ccc(F)cc2)n1)CC(F)F C(=O)(N=c1ccnc(Br)[nH]1)c1cccc(-c2cc(OCCCC)c(O)cc2C)c1 C(=O)(CC1COc2ccccc21)N(C)CC1CCCN1C(C1COCCO1)=O c1(NC(CC=C)C)ncc(C)cc1S(=O)(=O)NC1CCCC1(C)C C(CN=C(NCc1ccnc(OC(F)F)c1)NCc1ccco1)OC(C)C N1(C(CSCC)=O)CCCC(C2CC2NC(=O)C(F)OC)C1 C1(C(N)=O)CCCN(C(=O)CC2CCCN2Cc2ccc(C(=O)O)cn2)C1 C1(NC(C2CC(NC(CSCCN(CC)CC)=O)C2)=O)CCCCNC1=O N1(C(C(C=C)OC)=O)C2COCC1CC(NC(=O)CC1CC(F)(F)C1)C2 Cc1ccc(C(C)(C)C(=O)NC2CCC(N(C(=O)CCC3(C)CC3)C)C2)cc1 Cc1cccc(C=CC(N2CC3CC3(CNC(c3c(Cl)nn(C)c3Cl)=O)C2)=O)c1 N1(C(C(CCC)CNC(C2C3CCC(F)C23)=O)=O)C(C)CC2CCCC12 c1(C(=O)NC(CC2CN(C(C(CC=C)N(C)C)=O)C2)C)cnc2c(n1)CCCC2 O=C(CS(=O)(=O)CCCCO)NCCCCNC(c1cc2cc(F)ccc2[nH]1)=O C1(C)(C(N(CCC(N2CC(OCC#C)C2)=O)C2CC2)=O)CCCN1C c1(OC)ccc(Cl)c(C(=O)NC2CC(F)(F)CC2NC(=O)C=C(C)C(F)F)n1 C1(NC2C(C)CN(C(=O)OC(C)(C)C)C2)CN(c2ccccc2)CC1(C)C N1(C(c2ccoc2Cl)=O)CC(C2CCCN(C(C3CCC4CCC3O4)=O)C2)C1 C(C)(C(=O)NC1CC1C(c1cccs1)NC(=O)CSC)(C1CC1)OC C(C1CCOCC1)=CCN.CC(CSC(F)(F)F)C(=O)N1CC(n2cc(CS)nn2)C1 c1(C(N2C(CNC(C(=O)NCC)=O)COCC2)=O)cc(F)c(F)cc1I C1(CCNC(C2(SC)CN(C(C3CCCC3CN(C)C)=O)C2)=O)CCCC1(C)C c1(N2CC3CCN(C(CC(=O)OC)=O)C3C2)ncc2c(ccn2C)n1 c1(C(=O)NC(C#C)C(C)C)nnn2c1CSCC2 c1(C(=O)NCC2N(C(CC3CC(=O)C3)=O)CCC2C2CC2)cc2cc(Cl)ccn2n1 c1(C(=O)NC2CCCC(NC(c3c(C)ocn3)=O)C2)ccc2nnn(O)c2c1 N1(C(C(CC=CC)CC)=O)CC2(CCN(C(c3cnnn3CC)=O)CC2)C1 N1(C(c2nccc(OC)c2OC)=O)CCC2CN(C(=O)CCCCC#N)CC12 C1(C(=O)NCC(=C)C)CC(CNC(C2CCSC2)=O)C1 c1(NC(NCC(=O)NC)=NCCSC)ccc2c(c1)CCC2=O CCCCC(C)CCC(=O)N1CC2CCCC2C1C(=O)NCC1C(C)C1C C(CCC(F)(F)F)NC(C)CC1CN(C(=O)C=CC(=O)N(C)C)C1 c1(OC)cc(F)cc(C=CC(=O)NC2CCN(C(C3CC(C)=NO3)=O)CC2C)c1 C1(CC)CN(C(c2cc(C3CC3)n(C)n2)=O)CCN1C(=O)CSC1CC1 N1(C(C(C)C2CCC2)=O)CCCCC2(C1)CN(C(C1(CO)CCCC1)=O)C2 Cc1cc(C(=O)N(C2CN(C(c3sccc3Br)=O)CC2O)C)oc1C c1(OC)cc(Cl)sc1C(N1CCC1C(=O)Nc1ccccc1C(C)(C)O)=O C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC(C1CCN(C(C2(CCF)CC2)=O)CC1)C Cc1c(F)ccc(C(=O)NC2CC(C)(NC(=O)Cc3cccc(Cl)c3)C2)c1F c1(OCC)cc(CNC(=O)CCOC(C)(C)C)ccc1C N1(CC(=O)NCC(C)N(C(C2CCCCC2(F)F)=O)CC)CCC(=O)NC1=O N#Cc1csc(CNC(c2sccc2NS(=O)(=O)CC2CC2)=O)c1 N12Cc3n[nH]cc3C1C(=O)NCc1nc(co1)C2=O.C1(CC)(SC)CC1 Cc1sc(C)c(C(=O)NC2CCCC2NC(=O)C2=CCSC2)c1C#N N1(C(C=Cc2ccc(C)cc2)=O)C2CCC1CN(C(=O)CC1CC1C(F)(F)F)C2 n1(CC)cc(C(N2CCCC2CN(C(=O)C(F)(F)c2csc(C)c2)C)=O)cn1 Cc1nnc2c(C(N3CC(CNC(C4(C(F)F)CC(F)(F)C4)=O)C3)=O)cccn12 C1(N(C(=O)CC2CCC(=O)N2C)CC)CCN(C(=O)CCc2csc(C)n2)CC1 N1(NC(CN(C)C(C2(O)CCC2)=O)=O)CCC(n2cc(CCC#N)nn2)C1 O=C(C1COc2ccc([N+](=O)[O-])cc21)N1CC2(CCN(C(C3(Cl)CC3)=O)C2)C1 Cc1ccc(C)n1CC(N1CC2CC1C2NC(C1CC1Cl)=O)=O C(CCCC(F)(F)F)NC(C(C(C)NC(=O)CSC1CC1)C)=O CCC(C)(CNC(C1CC1c1ccco1)=O)NC(=O)CCc1cnccn1 CC1(CNC(C2C=CC=CC=C2)=O)CCCN(C(C2(CO)CCCO2)=O)C1 c1(Nc2ccc(SC)cn2)nc(C(=O)OC(C)C)ncc1Br N1(C(=O)OC(C)(C)C)CC2CC(OC(F)(F)F)CC1C2.C1(=O)C(C)(C)CCN1 C(=O)(C1Cc2ccc(F)cc21)N1CCC(NC(C(c2ccc(C)s2)C)=O)C1(C)C CCCCCCC(C)CC(=O)NCCC1CSCCN1C(c1cnnn1CC)=O O=C(C#CC1CCC1)NCC1CC(NC(C2CC2Cl)=O)C1 c1(C(N(C(C)C)CCN(C(=O)CCNC(=O)C=CCl)C)=O)ncccc1F c1(CC)cc(N2CCOC(C)(CNC(c3ccc(=O)n(C)c3)=O)C2)nc(C)n1 Cc1ccc2[nH]nc(CN3CCCCC(NC(c4cncc(Cl)c4)=O)C3)c2c1 N1(C(CSSC)=O)CCC2(COC(CNC(=O)Cc3cn[nH]c3)C2)C1 C1(N(C(C(C)CS(C)(=O)=O)=O)c2cnc(C(C)(C)C)nc2)COC2(CCNCC2)C1 CC(C)CC(C(C)(C)C)NC(=O)Cc1cnc(C(F)(F)F)s1 C12CCCC(C1)C2=O.N1(C(=O)NC(=O)C2CC2)CC2CC1C2C(F)(F)F CC(C)C(CC(=O)N(C1COCC1(C)C)C)NC(c1ccn(C2CC2)n1)=O c1(C(N2CCN(C(c3c(C)nc(Br)cc3)=O)CC2)=O)ccc(S(C)(=O)=O)c(Br)c1 C(CC)(C(=O)N1CC(CNC(=O)Cc2csc(S)n2)(COC)C1)OCC c1(C(N(CCCCCCNC(C(CCC)O)=O)C)=O)ccc2c(c1)N(C)CC2 C(c1ccc(C)cc1)=CC(=O)NCC1(CNC(CC(CC)OC)=O)CCC1 C#Cc1cccc(C(=O)NC2CCCN(C(=O)C(CC)C(=O)OC)C2)c1C c1(OCC)cc(C(=O)N(CC(CC)NC(=O)CO)C)ccc1[N+](=O)[O-] C1(NC(C2CCCC3(CC3)C2)=O)CCCCCC1NC(C12CCN(CC1)C2)=O Cc1nccc(CCC(=O)NCC2CC2CNC(=O)C(C)OC2CCCCC2)n1 N1(C(C(CC=CC)C)=O)CCN(C(C2CCN(CC)C2)=O)CC1C C1(CNC(c2cc3sccc3s2)=O)C2CCC(C2)N1C(=O)CC1CC=CCC1 c1(C(N2C(C)CC(CNC(CN(C(C(C)C)=O)C)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(CC(COC)NC(=O)CC(C)O)=O)CCCNC(=O)C1 C1(C(CNC(c2ccc(CC)s2)=O)C)CCN(C(=O)C(C)NC(=O)NC)CC1 C1(NCCn2ncc(CC)c2)CCCN(C(C2CNC(=O)C2)=O)C1CC N1(C(c2c(C#N)cncc2)=O)CC2CCC1CN(C(=O)CSC(F)F)C2 C1(CC(=O)NC2(CC=C)CN(C(=O)CCCC3CCC3)C2)CC2(CCCC2)CO1 C1(C(c2n(C3CC(CC)C3)nnn2)(CC)N)CCCC(C)(C)C1.c1(S)ccccc1 CCCC(C)(C)C(=O)N1CC(CNC(c2cc(C(C)(C)C)ccc2N)=O)C1 C(=O)(CCC(C)NC(=O)C(F)CCC)NCCCN(CCC)CC c1(CC(=O)NC2(CCNC(c3cc(CC)c(C)s3)=O)CCC2)c[nH]c(=N)nc1O c1(C(=O)NCC(CNC(C2(COC)CCCC2)=O)CO)cccc(Cl)c1 N1(C(CC=C(C)C)=O)CCCC2(CNC(c3cnc(C4CC4)s3)=O)CCCC12 Cc1c(C)c(C)c(C(N2CCCCCC(NC(C3CCCO3)=O)C2)=O)c(C)c1C Cc1cnc(C(N2CC=CC(NC(C3COC(=O)N3C)=O)C2)=O)c(C)c1 C(C(C)(C)C(=O)NC1CN(C(=O)C=CC2CCCO2)CC1COC)OCC N1(c2nnc(CC)s2)CCC2(CCCC2NC(c2ccc(F)c(F)c2)=O)CC1 CCC(C(=O)OCc1nc(C)c(-c2ccccc2)s1)C(C)C N1(C(CC)=O)CCCN(C(C2CN=C3N=CNN3C2)=O)CC1C C1(CNC(COCCC=C)=O)C2CC1N(C(=O)Cc1sc(C3CCC3)nc1C)C2 c1(-c2cc(CS(=O)(=O)N(C3CCN(S(=O)(=O)C)C3C)C)no2)ccc(Cl)cc1.CCO C1(C(=O)NC(C2CCCC2)CNC(C2(C3CC3)CCCO2)=O)(CC)CC1(F)F c1(N)cnn(C)c1.c1(CN(C(CNC(C(c2cnn(C)c2)C)=O)=O)C)ccccn1 N1(C(CSCCCC)=O)CC2CN(C(=O)CC3CC=CCC3)CC12 c1(OCCC)cccc(CNC(=O)Cn2cc(Br)c(=N)[nH]2)c1OC C1(C(=O)OC)CS(=O)(=O)CCN1C(C1C2CCCCC12)C(=O)NC1CCC1 C=CC(C)(CCOC)C(=O)N1CCC(C2CCCN2C(c2cnco2)=O)C1 N1(C(C(C)(C)C#N)=O)CCCC2(NC(c3ncccc3F)=O)CC2C1 C1(C(N2CC(O)(C(CNC(CCOCC)=O)(C)C)C2)=O)CCN(CC(F)F)CC1 C1(COC)(NC(=O)C(C)C2CCC2)CCN(C(c2cnccc2Br)=O)C1 N1(C(c2c(C(C)(C)C)c[nH]c2)=O)CC(NC(c2ccsc2CO)=O)C2(CCC2)C1 C(CCC(C)C(=O)NCCC(C)NC(=O)C(c1ccc(F)cc1)CO)OC CCC(C)C(C(=O)N1CCC(C(=O)NCCOC(F)(F)F)C1(C)C)N(C)C c1(CCC(=O)NCCCOCCNC(=O)C=CC=C(Cl)Cl)cc(Cl)no1 CC(C)CCCOCC(N1CCC(OCCNC(=O)CC2(C)CCCC2)C1)=O c1(OC)cc(C(N2CCCCC(CNC(C3CCCC(=O)N3)=O)C2)=O)cnc1Cl N1(c2n(CC(CC(C)O)O)nnn2)CCC2(CC1)CC(C(=O)OC(C)(C)C)=NO2 CCC(CC(C)C)C(=O)N(CCC(=O)NCC(O)C(F)F)C(C)C C1(CNC(C(CC)C)=O)CN(S(=O)(=O)Cc2ccc(F)cc2)CC(F)(F)C1 C1(CC(C)C)C(=O)NCCC(=O)NO1.C(C)(CCCO)NC(C)=O C#CCC(C)(CC)C(=O)N1CCN(C(C2CCN(c3ccccn3)CC2)=O)CC1 C(C)(C)(CC(=O)OC)N(C1CCN(CC)C1)C(=O)Cn1cnc(C(=O)OC)c1 c1(C(=O)NCC(C)NC(c2nocc2C2CC2)=O)c(O)nnc2c1CCCC2 c1(CC)nn(C)c(CC)c1C(N1CCCC(CC)(NC(C2CC2CC)=O)C1)=O c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CCC2)c(C)cc(Cl)cc1C C(=O)(C1CNc2ccccc21)N1CCCC(CNC(=O)Cc2ccc(O)nn2)C1 C(=O)(C(C(=O)NCC1(CC2CCC2)CC1)OC)OCC.C1C(N(C)C)CC(=O)N1 C(c1c(F)cccc1F)=CC(=O)NC1C(C)(C)CN(C(C2CCC2(C)C)=O)C1 c1(CNC(CSc2nc(C)[nH]n2)=O)cccc(NC(=O)COCCCF)c1 S(=O)(=O)(c1cc(C=CC(=O)NNC(=O)N=O)ccc1OCC)CCCN(C)CC C(CCC(=O)N=c1nc(C)[nH]c(OC)c1)=CCCC C1(NC(CC(CC)O)=O)CCC2CN(c3ncnc(C)c3OC)CCC2C1 Cn1cnc2nc(=NCCn3ccnc3Br)[nH]c(N3CCC(CF)C3)c12 C1(C(=O)NC2CCN(C(C(C)C3CCCC3)=O)C2)CCC(CCO)CC1 CCCCCCCCCC(=O)NC(CNC(C1CC(C)(C)CN1C)=O)CC C(=O)(CCCC(N)=O)NCCC(C)(C)NC(C1CC(C(F)F)C1)=O c1(C(=O)NC(C(C)NC(c2c(SCC)nccn2)=O)C)cc(C)c(Cl)c(C)c1 C1(CC)CN(C(c2cnoc2C)=O)CCN1C(=O)COCC(C)(C)C CCCS(=O)(=O)CC(=O)NC12CCN(C(=O)CN(c3ccncc3)C)CCC1C2 N1(C(C(=O)NCC=C)=O)CCC(CC(=O)OC)C(CC)C1.C1(=O)C(O)N1 N1(C(c2c(C)nccn2)=O)CCC2CC2(C(=O)Nc2ccc(CCO)cc2)CC1 c1(C(=O)NCC(C)(CO)NC(CCCCC=C)=O)nc[nH]c2nccc1-2 Cc1ccc2c(n1)CN(C(C1CCCCCN1C(C1CC(O)CN1C)=O)=O)C2 C1(CNC(=O)Cn2ncnn2)COCCN(C(C2(C(F)F)CC2(F)F)=O)C1 c1(C(N2CC(NC(CC3CCCC(C)C3)=O)C(C)C2)=O)cc2n(n1)CCC2 N1(C(c2cc(C)nc(O)n2)=O)CC2(COC(CNC(c3ccncc3Cl)=O)C2)C1 C(=O)(N=c1ccn(Cc2ccccc2OC(C)COC)[nH]1)NC(CC)(F)F C1(NC(C(C=C=C)C)=O)CC2CCC1CC2NC(c1ccc2c[nH]nc2c1)=O C12(C(=O)NC(C(C)NC(COCC(C)C)=O)C)CC3CC(CC(C3)C1)C2 c1(C(N2CCC(C(=O)NC(CCC(C)C)C)(C(C)C)C2)=O)cccn2ccnc12 c1(OC)nc(C)ccc1C(=O)NC1CC(CNC(C2C(C)CC2C)=O)C1 C(=O)(CC(C)(C)CC(=O)N(C)CCOCCC(=O)N(CCCO)CCO)OCC C(C(CC)(CC)C(=O)N1CCC(OCCF)C1)NC(C(C=C)(F)F)=O C(C(CO)C(C)C)NC(C(C1N(C(C(C=C)OC)=O)CCC1)(C)C)=O c1(C2C(C(N(C)CC3C4CN(C(C=CCOC)=O)CC43)=O)C2)cccc(Cl)c1F C1(NC(C2C(C)(CC)C2)=O)CCSC12CN(C(c1cc3n(n1)CCC3)=O)C2 c1(C(=O)NCC=CCNC(C2CCC2F)=O)ccnc2ccc(Cl)cc12 N1(C(=O)COCC(F)F)CCC(CF)(NC(C2CC(=C3CC3)C2)=O)C1 c1(N2CCC(c3scc(C)n3)C2)cc(=NCC(C)(C)CC2CC2)[nH]c(CO)n1.CC C1(C(N(CCNC(C2CC(SC)C2)=O)C)=O)CCCOCC1 C(CNC(=O)C1=NN(C)C(=O)CC1)(C(=O)N(CCO)OC)OC N1(CC(N2CC(C(=O)NC(CC=C)CO)(SCOC)C2)=O)C(=O)CNC1=O CC1CC=CCC1C(=O)NCC(CO)NC(c1cc(CO)[nH]n1)=O C(CCC(C)(C)NC(=O)CNC(C1CCOCC1)=O)NC(c1ccc(SC)s1)=O N1(c2ccnc(N(CCCn3ccnc3)C)n2)CCc2nc(O)c(C#N)cc2C1 C1(C(N(C)CC2(NC(CCc3cc(C)on3)=O)CC2)=O)CC(C)(C)C1C(F)(F)F C=CC(C(=O)NCCCOCCNC(C1CCS1(=O)=O)=O)OC N1(C(c2c(OC)scc2)=O)CCCC(CN(C)C(c2cn(CC3CC3)nn2)=O)C1 O=C1CC(C2CC2)(C(=O)NC2CCN(C(=O)C=Cc3cncs3)CC2CO)C1 N1(C(C2C(C)OC(C)C2C)=O)CC(NC(C2CC23CCOC3)=O)CC2(CCC2)C1 c1(C(N(CCCOC(C(C)OCC2CC2)=O)C)=O)cn2ncccc2n1 c1(C2C(C)CC2)nc(-c2ccncc2)nn1Cc1cccnc1 c1(C(=O)NC2C(NC(=O)COCC3CC3)COCC2)ccnc(Cl)c1O C1(O)(CNC(=O)C(O)Cn2cncn2)CCN(C(C2CC(F)(F)C2)=O)C1 C=C=CC(C)C(=O)N1CCC(C2CCCN2C(c2cnc(O)o2)=O)CC1 C(=O)(CC(C)(C)C(=O)N1CCCC(NC(C2CC=CCO2)=O)C1)OCC C1(CC)CC2CCN1C2=O.C(CCC(O)CO)NC(=O)COCP(C)(C)=O N1(C(COCC(C)(C)C)=O)CC2(NC(=O)CSCC(N)=O)CCC1C2 Cc1cc(C(N2CCN(C(C3CCC3)=O)C(C(C)C)C2)=O)c(C)n1-c1ccon1 C1(NC(=O)C=CCF)CCN(C(=O)CSC(F)F)CC1CC1CC1c1ccccc1 Cc1scc(C(N2CCC(C(N3CCC4CC34)=O)(CO)C2)=O)c1C Cc1nc(CNC(=O)CC2CN(C(C3CN(C4COC4)C3)=O)C2)oc1C c1(CC)nc(NC(=O)C(=O)Nc2ccc(OC)nn2)sc1C c1(C(CC(=O)OCC)NC(=O)NC(C)CC(=O)NC)ccc(Cl)cc1 C1(NC(C=CC=CC)=O)COC2(CCN(NC(C3(C)CCC34CCC4)=O)CC2)C1 c1(C(=O)NCC2CCN(C(C3=CC(C)(CC)C3)=O)CC2O)c[nH]c2ncccc12 N1(C(c2nccc(C)n2)=O)C2CCCC1CC(NC(c1cncc(F)c1)=O)C2 C1(CCC)CC(C(=O)N(CC(=O)NC2CC2COC)CC)C1 C=CC(C)(CCOC)C(=O)N(CCCCNC(=O)C(n1nc(C)cc1C)C)C CC(C)C(C(O)C(F)(F)F)NC(C1CN(C(=O)C=Cc2cccs2)CCC1O)=O C(=O)(CC1=NNC(=O)C1)NCc1c(CCNC(=O)C2=CCCCO2)ocn1 C(C1=NOC2CN(C(C3(CC(F)F)CC3)=O)CC12)NC(C(CC)CC)=O N1(CC(CCC)C)C(C(=O)OC)CC2CCCC12.N12CCCC1C2=O C1(CCOC)CN(C(=O)C(C)O)CCN1C(c1cnn(CC(F)(F)F)c1N)=O c1(NC(CSC)=O)ccc(S(=O)(=O)N(C(=O)Nc2nc(O)n[nH]2)C2CC2)cc1 CCC(C)C(CC(=O)NCC1(CC2CC2)CC1)NC(=O)CCC(C)N(C)C N1(C(C(C)CN2CCOCC2)=O)CC2CC1CC2NC(c1ccncc1F)=O N1(C(c2c(CC)nn(C)c2)=O)C(C(=O)N(C(C)CCC(C)C)C)CC2CCCC12 N1(C(c2ccc(CCC)c(N)c2)=O)CC(C)N(C(=O)CSC)CC1C C(=O)(CCC(=O)OC(C)(C)C)NCCN(C(=O)Cc1ccsc1Br)C(C)C C=C(COc1ccc(Oc2ccccc2)cc1)c1cccc(F)c1 c1(SCC(=O)NCC2C(NC(CSc3n(C)cnn3)=O)C2)ccc(F)cc1 C1(N(C(c2c(C)cc[nH]2)=O)C)CCC2CN(C(c3ccsc3)=O)CC12 c1(C(=O)NCC2N(C(C=CCOC)=O)CCCC2C)[nH]nc2c1CCC2(C)C C(=O)(C(=O)CC(C)C)NCC(C)(C(C)C)NC(c1c(CC)c[nH]n1)=O CC1=CCSC1C(=O)NCC(c1ccccc1)CNC(=O)COc1ccsn1 CC1=C(C(=O)N2CC(NC(c3scnc3C(C)(C)C)=O)CC2C)C(=O)OC1(C)C C1(C(=O)NC(C=C)CO)CCCN(C(=O)C(C(C)CC)OC)C1C C1(CNC(C2CC2F)=O)CC2CCC(C1)N2C(c1ncccc1C(F)(F)F)=O C(=O)(C#CC1CCOC1)NC1(CC)CN(C(c2sc(=N)[nH]c2C)=O)C1 C1(NC(C2C(C)OCCC2)=O)CCN(C(c2ccc(CN(C)C)o2)=O)C1(C)C C1(NC(C=C(COC)C)=O)CC=CCC1C(N1CC(OC(C)=O)C1)=O c1(C(=O)NC(CNC(C2CC(C)CC(C)C2)=O)C(C)(C)C)cc2c[nH]cnc-2n1 N1(C(C2CCN(C(c3c(CC)cns3)=O)C2C(C)C)=O)CCC12CCSCC2 c1(C(CNC(CN(C2CCCC2)C)=O)(C)C)ccn(C)n1 CN1C(=O)N(C)C2(CCN(C(C3CCCN3CC(F)(F)F)=O)C2)C1=O c1(CC(=O)NC2CC2CNC(C2CCC(=O)NC2)=O)c[nH]c2cc(F)ccc12 CCC(C(=O)N1CC(C)N(C(=O)C(CN(C)C)N(C)C)CC1C)C(F)(F)F c1(C(C(=O)NC2CCOC2)N(C2CC2)CC)cc2cc(Cl)ccc2s1 C(=O)(C1CCCc2cccnc21)N1CC(NC(CCCCC)=O)C(CO)C1 N1(CCOC)CCN(C(c2ncc(C)s2)C(=O)NCCC2(C)CC2)CC1C CC1CN(C(C)C(=O)Nc2cccc(F)c2)CCC1NC(c1cc(C2CC2)no1)=O CC1(C)CC(C(N2CC(F)(CO)C2)=O)CN(C(=O)COC2CCCCC2)C1 C1(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)CN2CCCN1CC2 N1(C(c2cnn(CCC)c2C)=O)CCN(C(c2ccoc2CC(N)=O)=O)C2CC12 c1(C(N2CC(CCNC(C(CCC)O)=O)C(C)C2)=O)cc(C)c(C)nn1 N1(C(C(C)NC(C)(C)C)=O)CC2CCN(C(=O)CNS(=O)(=O)N(C)C)C2C1 c1(C(C(=O)N(C(C)C)CCNC=O)C)ccc2c3c(cccc13)CC2.C1CC1 CC(CCN(C)C(C1CCOC1)=O)NC(=O)CCc1cncs1 Cn1cnc(C(N2CCCC2CCNC(c2cncc(C(N)=O)n2)=O)=O)cc1=O c1(C(N2CC(O)CC(NC(C=NOC)=O)C2)=O)c(C)nc2sccn12 CC(C)(C(=O)NCC1CC1NC(=O)CCCOc1cccnc1)c1ccccn1 c1(OC)c(Cl)cc(C(=O)NCC2CCC(C)(C)C2)c2ncccc12 c1(CC)cnccc1C(N1CCC(C(=O)NCC(O)CC(C)C)CC1)=O c1(C(N(CCC(C)NC(=O)CCCCC2CC2)C)=O)c(Cl)ccc2c[nH]nc12 c1(CCC(=O)NCC(CNC(CCC=CC)=O)OC)cccnc1Br C1(NC(C23CC(C)(C2)C3)=O)CCOC12CCN(C(=O)C1=CS(=O)CCC1)CC2 c1(CC(=O)NC(c2nccs2)(C)C)cccc(S(=O)(=O)N2CCCC2)c1 C1(C(=O)NCCCCOCCNC(C(C(C)C)NC(C)=O)=O)COCC(C)(C)O1 c1(CC(=O)NCC(C)CN(C)C(C2CCCCCC2)=O)ccc([N+](=O)[O-])c(N)c1 c1(N(C23CCC(N)(CC2)C3)C(c2cc(C)[nH]c2)=O)nc(C)nc2c1CCC2 CN1C(=O)CCC1C(=O)NC1C2CC(NC(c3ccn(C4CCC4)n3)=O)CC12 CCCCC(C(=O)NC1(C2CN(C(C3(N=[N+]=[N-])CC3)=O)C2)CC1)C(C)C Cn1cnc2ccc(C(N3CCC(CCNC(C4CCCO4)=O)CC3)=O)cc12 Cc1cccc(C(=O)NCCCCCC(=O)NC2CCCC2F)c1C Cc1c(C(=O)N(CCC#N)C2CC2)[nH]c2cc(C(=O)NC3CCCC(C)C3)ccc12 N1(C(CC(=C)C)=O)CCC(NC(=O)C(C)(C)C2CCOCC2)CC1C Cc1c(C(=O)NC(C(N)=O)C(C)(C)C)[nH]c2ccccc12 c1(OC)ccncc1C(=O)NCCCN(C(=O)CCc1nc(C)cs1)C c1(CNC(C=CCN(C(=O)CC2CC2C(F)(F)F)C)=O)ccn2ccccc12 C(=O)(C#CC1CCCC1)NCC1CC(OC)CN1C(=O)C=Cc1ccn(C)c1 Cc1cc(C(=O)NC2(CNC(=O)COc3cnn(C)c3)CCC2)c2nccn2c1 CCC(C)(CCC(C)C)C(=O)N1CCC(CNC(c2ccc(O)c(F)c2)=O)C1 N1(C(C(C(=O)OCC)c2ccccc2)=O)CC2CCC(C1)N2C(=O)CS(N)(=O)=O c1(C(=O)NCC(=C2CN(C(CSSC)=O)C2)F)ccc(=O)n(O)c1 CS(=O)CCC(=O)NCC1(O)CC(CNC(C2CC(N(C)C)C2)=O)C1 N1(C(C)C(=O)Nc2cc(Cl)c(Cl)cc2Cl)CCC(N(C)C)CC(C)(C)C1 C1(Cn2cc(N(CC)CC)c(-c3ccccn3)n2)CCCCC1(C)C C1(CNC(c2cnc(C(C)C)s2)=O)CC(NC(=O)CC2C(C)(C)C2(C)C)C1(C)C C(N=c1[nH]n(C)cc1[N+](=O)[O-])C1C(C)CCN(C(c2ncc(OC)c(C)n2)=O)C1 Cc1nnc(CC(=O)NCCOCCCN(C)C(c2ccnn2C(F)F)=O)s1 C12CCC(C)(C)CN1C2.c1(CCCCCNC(C(CC)SC)=O)ccccc1Cl C1(C)(NC(c2c(CC)ccs2)=O)CCN(c2nnc(C(C)(C)C)o2)C1 C(C(C(C)C(C)C)NC(c1coc(C(F)F)n1)=O)NC(CC(=C)Br)=O c1(C(N2C(C)CC(NC(c3cc(F)n(C)n3)=O)C2)=O)cc(O)c2ccccc2c1 C(=O)(C1CCCc2ccccc21)N(C)CCOCCNC(C1CC=CC(O)C1)=O c1(C(N2C(C)C(NC(=O)CCC3CC(C)(C)CO3)CC2)=O)ccc2c(c1)CC2 N1(C(c2ccc(COC)o2)=O)CCOC(C(=O)NCC#CC2CC2)C1 S(=O)(=O)(c1cnn2ccc(N(C)CCOC)nc12)NCC1CC(=C)C1 C1(OC)CN(C(=O)C(F)CC2CCOC2)CC1NC(=O)C(CSC)CC1CC1 C(=O)(C(C)CC(=O)c1ccccc1F)NC(C(C)NC(Cn1cc(C)nc1)=O)C c1(C(=O)NC2CN(C(C3(CC)CC3(F)F)=O)CC2F)c(F)cc(F)cc1F c1(NC(C2N(C(C3C(C)C3)=O)CCCC2)=O)cncc(C#N)n1 C1(C(=O)NCC2OCC(C(N(CC(N)=O)CC)=O)C2)CCCC(C)C1 CC(C)C(F)(F)CC(=O)N(C(c1ccccc1)CNC(C1CC(CCO)C1)=O)C C(CS(=O)(=O)CC(=O)NCCN(C(=O)C(=O)N=S(C)(C)=O)CC(C)O)OC Cc1cc(C(N2CCCN(C(C3OC4CCC3C4)=O)CC2)=O)ccc1Br Cn1cc(C#N)cc1C(=O)NC1CC(F)(CNC(C2CC(=O)NC2(C)C)=O)C1 C(=O)(CCCC(=O)c1ccc(Br)cc1)NC(CC(=O)OC)c1cccnc1 C(=O)(C1=CC2CCC(C1)C2)NCC(CC(=O)NC(CC#CC)C)(C)C C1(O)(CNC(c2cc(C(N)=O)ncc2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1 c1(SC)cc(C)nc(N2CC3CN(Cc4ccc(N5CCCCC5)s4)CC23)n1 N1(C(CCCCC#C)=O)CC(CO)C2(C1)CN(C(=O)C(CCC)N(C)C)C2 C1(C(N(C)Cc2c(C)ncs2)=O)CCC(C(C)C)N1C(C1CC1CCN(C)C)=O N1(C(C2(CC=C)CCCC2)=O)CCCC(CNC(=O)Cc2csc(NC=CC)n2)C1 CC1(F)CN(c2ccc(S(=O)(=O)N3CCCC3C3CCCC3)cn2)CCC1O c1(CNC(=O)NCc2ccn(-c3ccc(Cl)cc3)n2)cnc2c(F)cccc2c1 c1(OC)cc2ccc(Nc3nc(-c4ccccc4Cl)no3)cc2cc1OC C(=O)(C(C#N)C1CC1)N(CC(=O)NCC1CCC1)C.C12(CC1)C(=O)N2 C1(NC2C(C#C)CCCC2)CC2(CCN(Cc3ccccc3)CC2)C1 N1(C(C(C)NC(=O)NC)=O)CCC(NC(c2cc(F)n(C)n2)=O)C(CO)CC1 C1(C(=O)NCC23COCC(C2)C3)CCN(C(=O)C(=O)N2CCCCCC2)O1 c1(C(=O)NC2C(NC(C3NC(=O)OC3)=O)CCCC2)cc(F)cc(F)c1 c1(CCC(=O)NC2C(OC)CN(C(=O)C3=C(C)CCC3)C2)ccc(Cl)c(C)c1F CCCCC(=O)C(=O)NCC(C)(C)CC1CN(C(=O)CC2CCCCC2(C)C)C1 Cc1sc(C(=O)N(C2CCN(C(C3CCN(C)C3=O)=O)C2)C)cc1[N+](=O)[O-] C1(C(N(CCC#C)C)=O)CC2CCC1N2C(C1(CC=C)CCOC1)=O N1(C(c2c(CCC)[nH]cc2)=O)CC(C)(C)CC1C(=O)N(C)CC1(C)CCC1 c1(CNC(C(n2cc(COc3cnn(C)c3)nn2)C)=O)nncn1C Cc1nc2cc(C(N3CC(OCCNC(=O)CC(C)c4ccco4)C3)=O)[nH]c2s1 c1(CC(=O)NCC(CCNC(CSCCN(C)C)=O)O)ccnc(F)c1 Cc1cc(C(=O)NC2(C(=O)NCCC3CCC(=O)N3)CSC2)nc(O)n1 N1(C(C2(CCC)CCC2)=O)CCCC(O)(CN(C)C(C2CCCO2)=O)C1 N1(C(C(C)OCCC(C)C)=O)CCOC(C(=O)NC2CCOCC2F)C1 c1(C(N)=O)ncc(NC(=O)C=Cc2ccc(-c3ccccc3F)o2)cc1F Cc1oc(C(C)C)cc1C(N1CC(NC(c2ccno2)=O)C(CC(C)(C)C)C1)=O c1(C(C(C)NC2CCN(C(=O)Nc3cn(C)cn3)CC2)O)c(Cl)cccc1Cl N1(C(c2c(=O)cc(C)[nH]c2)=O)CCC(C(=O)NCC(F)C(C)(C)O)C(C)(C)C1 C1(NC(c2c(CC)cccc2C)=O)CC2(C1)CC2N=c1ccc(C)n[nH]1 c1(C(N(CCN2CCN(C(C(CC#C)C)=O)CC2)C)=O)[nH]nc2cnccc12 c1(C(=O)OC)n[nH]c(=NC2CCN(C(C3(S(C)(=O)=O)CCCC3)=O)CC2C)s1 C(CC(O)C(=O)NCC1(CC(c2ccnc(OC3CCOC3)c2)=O)CCC1)SC Cc1[nH]c2ccccc2c1CC(=O)NC1CC1NC(=O)Cc1cncnc1O C(CS(=O)(=O)Cc1ccccc1)OC1(C)CCCN1 N1(C(C(C)(CC2CCC2)OC)=O)CC2(CC(NC(=O)Cc3cnns3)CO2)C1 CC1C(C(=O)N(CC(C)(C)C)C)CCN1C(=O)CN1CCC(N(C)C)C1 Cc1ccc(C)c(C(=O)NC2CC(CCNC(=O)C(O)C3CCCC3)C2)n1 N1(C(C(C)n2ccnc2)=O)CCOC2CCN(C(c3ccc(CO)o3)=O)CC12 N1(C(c2cnc(CC)o2)=O)CCCC(F)(C(N2CCC(O)C(O)C2)=O)C1 C1(CCNC(C(C)NC(=O)OCC)=O)CCN(C(c2ncoc2C)=O)CC1 N1(C(C2=C(C)CCCC2)=O)CCC2(CCOC2)C(CNC(c2cc(C)on2)=O)C1 C(CC(=O)Nc1ccccc1OC(F)F)(C(F)F)NC(c1cnn(C(C)C)n1)=O C1(CC(=O)NCCCC)CC(NC(=O)CCCNC(=O)OCC)CCO1 N1(C(C2CCC(C)O2)=O)CCC2(CC1)OC1(C)CC2(NC(c2ncccc2F)=O)C1 C1(NC(C2(CC)CC2)=O)CCCCN(C(c2nnsc2COC)=O)C1 CC(CCCNC(=O)CNC(c1ccccc1)=O)NC(=O)CN1CSCCSC1 Nc1c(C(=O)NCCC2CN(C(=O)CC3=NNC(=O)C3)CCO2)cc(Cl)cc1F C(=O)(C1=C(Cl)CCCC1)NCc1scc(CNC(C(CCOC)C)=O)n1 c1(OCC)cc(CO)ccc1C(N1C2CC1CN(c1ccnc(N(C)C)n1)C2)=O C1(C(=O)NC(CCN(C(COCC(=O)OC)=O)C)C)Cc2n[nH]cc2C(=O)N1 c1(C(C)=O)ccc(F)c(C(=O)NC(C)(C)C(C)NC(=O)C2=C(Cl)CC2)c1 C1(C)(NC(=O)NCC(=O)OCC)CCN(C(c2sc(Cl)nc2Cl)=O)C1 c1(-c2c(C(=O)NCC(CNC(CC3(C)CC3)=O)F)c[nH]n2)ccc(Cl)cc1 c1(CCC)nc(C)c(C(=O)NCC2(C)CCCN2C(=O)C(O)C(F)F)o1 c1(N(CCC)C)nc2c(c(=NCC3CCCCC3(F)F)[nH]1)CC(C)CC2 N1(C(C2N(C(COCCOC)=O)CCC=C2)=O)CCCN(C)CCC1 N(C(=NCCCCl)N1CCC(c2ccccc2)C1)CC1(CO)COC1 c1(NC(c2c(CNC(C(=O)NC)=O)cc[nH]2)=O)cc(C)c(F)c(C)c1 c1(NC(C2(C)CCCN(C(C(N3CCCCC3)C)=O)C2)=O)cnc2c(c1)CCC2 CC(C)C(C(C)NC(c1c[nH]c(=N)o1)=O)NC(=O)CNC(=O)C1CC1 c1(C(N2CC(CCNC(c3coc(C)n3)=O)(OC)C2)=O)cc(C(F)F)ncn1 C(=O)(CCCCC(N)=O)N1CC(CNC(=O)CCCN2CCCC2)CC(C)C1 c1(CCCSC)cn(C2CCC(C(=O)Nc3csc(C(O)C4CC4)n3)C2)nn1 c1(C(N2CCC3CN(C(C4C(=C)C4)=O)C3C2)=O)ccc2c(c1)OCCO2 C(=O)(C(C)(C)CN(C)C)NC(c1ccccc1)C(C)NC(c1c(CC)nco1)=O c1(COC)c(C(N2CC(NC(=O)CC(C)(C)C)C3CC3C2)=O)sc2ccccc12 C12(C(=O)NCC3(CO)CC(C)C3)CCC(CN(C(=O)CC(O)C(C)C)C1)C2 c1(CC(=O)NCC(CNC(C2(C)CCOC2)=O)(C)O)cnn2ccccc12 N1(C(c2ccc(CC)[nH]2)=O)CCN(C(=O)Cc2nnc(C)s2)C2CC12 C(CC(C)C)(C(=O)NOCCCF)NC(CCC(C)=O)=O N1(C(=O)Nc2n(C(c3cccc(Cl)c3Cl)C)ncc2)CC(C(N)=O)CC(F)(F)C1 c1(C(N(C2CCCCN(C(C(C)OC)=O)C2)C)=O)oc2ccccc2c1C N1(C(C(C)=C(C)C)=O)CCC(C)(C)CC1C(=O)N(OC)C(C)C C(=O)(CCCCc1cnn[nH]1)NC(C)C(CO)NC(C1CCCCCC1)=O Cc1nn(C)cc1C(C)C(N1CCCC1CNC(=O)Cc1cn(C)cn1)=O N1(C(c2ccc(C#C)nc2)=O)CC2CC(NC(=O)CC3CC(C)C3)C(C2)C1 CC1CN(C(=O)CCCF)CC(C)CN1C(=O)COC(F)(F)C(F)(F)F Cn1cc(Br)cc1CC(=O)OCc1cscc1-c1ccccc1 N1(C(C(C)NC(=O)OC)=O)CCC2(C=C(C(=O)N3CC(=O)CC3(C)C)C2)C1 N1(C(C(CN(C)C)NC(c2ncc(OC)nc2)=O)=O)CCCC(F)(CO)C1 C1(C)(CNC(C(C)C#N)=O)CCCN(C(c2ccc(Cn3cc(F)cn3)o2)=O)C1 N1(C(C(COC)C)=O)CCCCC1C1(CNC(=O)C(C(C)O)NC(C)=O)CC1 Cc1n[nH]c(C)c1SCC(=O)NC(C)C(C(C)C)NC(=O)CCn1ccnn1 c1(C(C)C)ccc(C(=O)NCC2CCC2NC(C2COC(=O)N2)=O)s1 N1(C(c2cc(C)n(C)c2)=O)CCCC2(NC(=O)CC(O)CC(C)(C)C)CCCC12 C1(N(C)C)CCC2(CC1)CN(S(=O)(=O)Cc1ccc(Br)cc1)C2 c1(OC)c(F)cc(C(=O)N(C2CCCC2)CCNC(C2CCCC2O)=O)cc1Br c1(C(=O)NCC(CNC(c2c(CC)cccc2F)=O)F)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)OC)cc(Br)c(NC(N2CCC(O)CC23CC3)=O)nc1C C(=O)(C1CCCc2ncccc21)NC1CCC(NC(C2C(C)(C(C)C)C2)=O)CC1 C(C(COC)CC(=O)NC1CN(C(c2ccon2)=O)CC1OC)OC c1(OC)ccnc(C(N2CCC(C(C)NC(=O)C(O)C3CC3)C2)=O)n1 c1(C(=O)NC(C(C)NC(c2c(Cl)ccc(F)c2F)=O)C)ccc(O)cc1[N+](=O)[O-] C1(CNC(C2C(=O)NCC2)=O)CCCCN1C(=O)CCOCC1CC1 Cc1[nH]nc2cc(C(=O)NC3(CCNC(C4SCCC4C)=O)CCC3)ccc12 c1(C(=O)NCCCN(C(C=CC(C)C)=O)CC2CCCC2)csc(C(C)(C)C)c1 c1(NCC(CC(C)C)NC(c2ccnc(F)c2)=O)cc(C#N)c(F)cc1[N+](=O)[O-] CCCC(CCC)CC(=O)NCCC12CCC(C1)N(C(=O)CC(C)SC)C2 C(=O)(C(C)(C)CC(F)(F)F)NC1C(CN(C(c2cc(C)nc(O)n2)=O)C)CCC1 N1(CC(=O)NCC23N(C(Cc4cn(C)nc4)=O)CCC2CC3)C(=O)CC(C)(C)C1=O N1(C(c2cc(C)c(Cl)cc2)=O)CCC(C2CCCN(C(=O)C(C)NC=O)C2)C1 C(=O)(C(C)CC(C)(C)C)N1CCC(C(=O)NCCC(=O)OC)(OC)C1 N1(C(CNC(C2CCN(CC)C2)=O)C)CCN(C(C2CCCS2(=O)=O)=O)CC1 C1(OCC(N2CC(NC(=O)CC(C)COCC#C)C2)=O)(CO)CC(C)(C)C1 C(=O)(C1=COCCO1)Nc1cccc(CC)c1.C12(OC)CCN(C1)C2=O c1(C(=O)NC2(CO)CN(C(C3C(C=C)OCC3)=O)C2)nccc2ncccc12 C(C(CC1CC1)C(=O)NCc1cn(C2CC2)nn1)NC(COC)=O C1(NC(CN2CCC(C)(O)C2)=O)(CO)CCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 N1(C(COC(C)C)=O)CCCC(CNC(=O)C(=Cc2c[nH]cn2)F)CC1 C12(NC(C3C(CNC(Cc4cc(COC)on4)=O)CCC3)=O)CCN(CC1)CC2 C(CC(O)N(C(=O)CNC(C)=O)C)N(C(CNC(=O)NC)=O)C.OC C1(NC(=O)CN2CSCC2=O)CN(C(=O)CC2CCCO2)C2(CCCCC2)C1 c1(C(N(CC(C)O)CCNC(C2CCCO2)=O)=O)cc(Br)cc(F)c1F C(=O)(C1=COCCC1)NC1(C)CC(NC(C2C3CNC(=O)C23)=O)C1 N1(C(c2ccc(CC)o2)=O)CCN(C(=O)C(F)CCC(C)C)CC12CC2 N1(C(C(C)N2CC(C)C2)=O)CCC(OCCNC(COCC2CC2)=O)C1 CC(C)CC(C(=O)NC1C2CCC1N(C(=O)CCOCCN(C)C)C2)C(C)C c1(CC(C)C)ccccc1C(=O)OC(C)(C)C.C12(CCSC1)CN(C)C(=O)N2 c1(-c2ccnc(SC)n2)nc(C(=O)Nc2cnn(C)c2)n2ccccc12 c1(C(C(=O)NC2C(CNC(C3(COC)CCC3)=O)CC2)O)ccc(Cl)c(Cl)c1 CC1CCC(Cl)=C(C(=O)NCC2(O)CCCN(C(c3cc(Cl)cn3C)=O)C2)C1 c1(C(C)C)c(C(N2CC(F)(CNC(=O)C=C3CCN(C)C3)C2)=O)cnn1C N12C(CC3CCCCC13)C2=O.C=CCS(=O)(=O)N(C(C1CCC1)C)CC c1(C(N2CCC3(NC(c4cnc(O)o4)=O)C(C2)C3)=O)cc(F)c(F)c(F)c1F c1(C(=O)NCC(C)(Cn2cccn2)NC(c2coc(Cl)n2)=O)cc2ccncc2[nH]1 C1(NC(C2CC=CCO2)=O)C2CCC1N(C(c1cc(C3CC3)nc(O)c1)=O)C2 Cc1oc(C(C)C)nc1C(=O)NC1(CNC(C2CCCC(C)C2)=O)CCCC1 C1(CNC(=O)CC23COC(C)(C2)C3)CN(C(c2cnc(S)nc2)=O)CCC1N C(=O)(C1CCCc2scnc21)NC(CNC(c1coc(C(F)F)n1)=O)CO c1c(C(CCC2CCCO2)NC2CC2C2CCCO2)nnn1Cc1ccccc1 Cc1cccc(C(N2CC=C(CNC(=O)C(F)C3CCOC3)CC2)=O)c1F C1(N(C)Cc2cccc(N(C)C)n2)CS(=O)(=O)CC1O C1(C(N2CC(CC(C#C)C)C2)=O)(CC=C)CN(C(=O)C(c2ccnn2C)C)C1 N1(C(c2cccc(CC)c2)=O)CCC(C)C(NC(C2(CC(F)F)CC2)=O)C1 CCC(C)(C(=O)N(C)CCOCCNC(c1cccc(F)c1O)=O)C(N)=O C(=O)(C1CCCc2cncn21)NCCOC1CCN(C(c2c(N)cn(C)n2)=O)C1 C1(CC)(NCc2c(F)cncc2F)CCN(C(=O)OC(C)(C)C)CC1 N1(C(C(CCC)(C)O)=O)CC2(CC(C(N3CC(C(C)(C)O)C3)=O)CO2)C1 c1(OC)cccc(NC(C2CCC2(F)F)=O)c1Br C(CCCCC(=O)O)(C(=O)NC1(C(=O)OC)CC1)N(CCC)CCC c1(C(=O)NCC2CCN(C(CCCC(CC)C)=O)CC2)cc2cccn2c(O)n1 CC1CCC(=CC(=O)NCCC(C)NC(=O)CSC(F)F)C1 C=CC(C)(CCOC)C(=O)NCC1COCC1NC(=O)CCc1cc(C)no1 c1(N2CCC(NC(CN3CC(=O)NCC3)=O)C(F)C2)ccnc2ncnn12 CC1(C)OCCOC1C(N1CC(NC(=O)CCCC(N)=O)CC(F)C1)=O Cc1c(NC(C)CC(=O)N(C)C)ncnc1N(C)Cc1ccsc1 CC(C)CCC(=O)NC1CCCCC1NC(C1CCC1)=O.C1(CN)CCC1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCCC(N(C(C(CC)CC)=O)C)CC1 C(CCC(C)C)=CC.C1(=O)CC=CC(=O)NCC2(CC2)CCN1 N1(C(c2nccc(C)c2)=O)CCC(F)(F)C(CNC(c2ccc(C)cc2F)=O)C1 CC1(C(N2CCC(O)(CNC(c3cscc3C(F)F)=O)C2)=O)CCNC(=O)C1 C1(NC(C2C(=C)C2)=O)CC12CCN(C(=O)CC1C=CCCC1)C2 Cc1ccc(F)c(N)c1C(N1CC=C(CCNC(=O)C(C)SC(C)C)CC1)=O C1(C(N2CC(F)(CNC(CN3CC(=O)NCC3)=O)C2)=O)CCc2nc(O)[nH]c2C1 c1(C(=O)NC2CN(C(CC(C)(C)O)=O)CC2C(F)F)cnc(O)c2c1NCCC2 CCC(F)(F)CC(=O)NCC(C)(O)CNC(c1nc(C)ccc1F)=O C1(O)(NC(=O)C(c2ccccc2)O)CCN(C(c2ccnc(OC(F)F)c2)=O)C1 N1(C(CC(C)F)=O)CCCC2CN(C(=O)C(=Cc3ccccc3)C#N)CCC12 N1(C(C2C(C)OCCC2)=O)CCC2CCC(C1)N2C(C1CN2CCN1C(C)C2)=O N1(C(COCCN(C(C2C(=C)C2C(=O)OC)=O)C)=O)CCC2CN(C)CC2C1 C1(CNC(C=CCCC)=O)CCN(C(c2ccc(Cl)c(C(F)F)c2)=O)C12CCC2 C(=O)(C(C)S(N)(=O)=O)NC1C2CN(C(C(C3CCC(=O)N3)C)=O)C1C2 C(c1ccccc1F)=CCC(=O)NC(CNC(c1[nH]cc2c1CCC2)=O)C1CC1 C(C)(C(=O)N1CCCC(NC(C2CC23CCOC3)c2nncn2C)C1)(C(C)C)OC C1(C(=O)NCCCN(C)CCO)CC2(CCOCC2)CN1C(=O)OC(C)(C)C c1(C(=O)NC2C(C(=O)NC(C#C)C3CCC3)CCCCC2)cc(C)cc(C#N)c1 Cc1cc2ccc(C(=O)NCCNC(c3ccc(F)c(SCC#N)c3)=O)cn2c1 N1(C(C(CNC(C2(C)CC2)=O)O)=O)CCCOC(C)(C)C1 CC12CC1CCN2C(C1C=CC(NC(C2CCCCO2)=O)C1)=O C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CC(N)=O)(NC(=O)CC2CC2)CC1 C1(NC(c2c(OC)nn(C)c2)=O)CC2CC1N(C(=O)Cn1ccc(C)cc1=O)C2 N1(C(c2c(C)cc(C3CC3)cc2)=O)CC2(CCCCN2C(=O)C2=CC(C)(C)C2)C1 N1(C(C=C(C)C(F)F)=O)CCN(C(=O)CCc2ccn(C)n2)CC1c1cn[nH]c1 CN1CCOC(C(N2CC3CC2C3C(=O)NCC2COC(C)(C)C2)=O)C1 c1(CNC(=O)NC2CCN(CCSC3CC3)C2)cc(-c2ccccn2)cc(F)c1 CC1(C)CCCN(C(c2ccc(F)cn2)=O)C1C(=O)NCc1ncc(Cl)cn1 CC(C)CCC(F)C(=O)N(C1CCCC1)CC(N1CCC1CN=[N+]=[N-])=O C1(CNC(C(CC)C(=O)OC)=O)COC(C)(C)CN1C(=O)CC(C)(C)CN(C)C N1(C(C2(CNC(=O)C(F)CC3CCOC3)CC2)=O)CCCC(F)C1 c1(C(N2CCC(NC(C3C(OCC)C3)=O)C2C2CC2)=O)c(C)cc(=O)oc1C C1(C(=O)N(C2CCOC(C)C2)C)(COC)CCN(C(c2c[nH][nH]c2=N)=O)C1 CCCCC(C(=O)NC1CCCC(C(=O)NCCN(C)C2CC2)C1)C(C)C N1(C(c2nccc(C(N)=O)c2)=O)CCC2(CC1)CC2NC(=O)CCCC1CC1 c1(C(N2CC(O)(CN(C(C(C)OCC#C)=O)C)C2)=O)cnn2c(C)cc(C)nc12 N1(C(C)=O)CCC(c2cccc(F)c2)C(NC(=O)CCCOc2ccccc2)C1 C1(NC(C(CC=C)C)=O)CN(C(C2CCc3nnc(O)n3C2)=O)C2CCCCC12 C1(Nc2nc(C)nc(N3CCOCC3)c2)CCOC2(CCSC2)C1 Cc1cccn2nc(C(N3CCCCC3CNC(C3CCS(=O)CC3)=O)=O)cc12 C(N=c1cc(CC2(CCOC)CC2)nc[nH]1)C1(C(C)(C)C)CCN(C=O)C1 c1(CSC)ccccc1C(=O)NCCOC1CCN(C(=O)CC2CNC(=O)C2)C1 C(=O)(C1=CS(=O)CCC1)NCC1CCC(NC(c2cnc(OC)c(Cl)c2)=O)CC1 c1(C(N(C2CC(NC(C3(F)CC3C)=O)C2)C)=O)cccc(C(F)(F)F)c1 N1(C(c2nc(C(C)C)oc2)=O)CCN(C(c2c[nH]c(C#N)c2)=O)CC(C)C1 c1(C(N(CC(CNC(C=C(C)Cl)=O)O)C)=O)nc(C)n(C)n1 C1(NC(c2nc3ncccn3n2)=O)CN(c2nccnc2F)CC2(CCC2)C1 C1(NC(C(C)=CC2CC2)=O)CC(O)CN(C(=O)CCOC2CC2)C1 Cc1nc(CC(=O)N(CCC(C)NC(c2ccn(CC(C)C)n2)=O)C)c(C)s1 CC(C)(C#N)CCCC(=O)NCCC1CC(F)(F)CN1C(c1cnsn1)=O C1(CNC(COC2C(C)CCCC2)=O)CN(C(=O)CC(F)(F)F)CC2(CCC2)O1 C1(CC(=O)OC)CC(NC(=O)CC2CCSCC2)CCO1 c1(C(N2C(C)CC(CNC(c3cc(Cl)cn3C)=O)CC2)=O)n[nH]c2c1CCSC2 CC1C(NC(=O)CSCc2ccncc2)CC2CCC1N2C(C1CC(F)(F)C1)=O c1(C(=O)NC(C2(CNC(C3OCCN(CC)C3)=O)CC2)C)nccc2occc12 C1(N(c2nccn2C(C)C)C(C2CN(C(=O)OC)C2)=O)CCNCCC1C CC1(C)COC(CC(=O)NC(CC2CCC2)C(=O)NCC2(C)CCC(=O)N2)C1 N1(CC2N(C(c3c(C)ccc(I)c3)=O)C3C(C2)C3)CCN(S(=O)(=O)N(C)C)CC1 C(c1cnn(C)c1C)=CC(N1CC(O)(C(CNC(COCCCC)=O)(C)C)C1)=O CCCC(CC)C(=O)N1CCC(C(F)CNC(=O)CC2(N(C)C)COC2)CC1 CCCCCC(F)C(=O)N(C(C)CNC(=O)CCC=Cc1ccccc1)CC CCC(O)C(=O)NC1CC(F)(CNC(=O)CCN2CCOCC2)C1 c1(NC(C)Cc2ccc(F)cc2F)nccc(=NC2CC3CC(OC)C3C2)[nH]1 C(=O)(C1=CCCN(C(=O)C(O)C(C)(C)C)C1)NC(C1(O)CCC1)C C1(C(N(CC(CN(C(COC(CC)(C)C)=O)C)O)C)=O)CC(F)(F)C1 C1(CNC(Cc2nc(C)[nH]n2)=O)CN(C)CCN1C(=O)C(=O)C(F)(F)F C1(C(=O)NC2C(CC)CN(C(c3cccc(C)c3O)=O)C2)CCc2nn[nH]c2C1 c1(C(=O)NC2CN(C(=O)Cn3cncn3)CCC2O)cnc2ccccc2n1 N1(S(C2C(C)OCC2)(=O)=O)CCC(N)c2cc(Cl)ccc21 C1(NC(C=C(C)C(C)C)=O)CS(=O)(=O)CC1NC(=O)C=Cc1ccccn1 Cc1ccc2[nH]c(C(=O)NC(C)CN(C)C(c3ccccc3C3CC3)=O)cc2c1 N1(C(c2c(C)con2)=O)CCN(C(=O)C(C)(C)C(=O)OC(C)(C)C)CC1CF C1(CC(=O)N(CC(C)NC(=O)C(F)(F)c2cnccn2)C)CCCS1(=O)=O N1(C(C(c2ccc(OC)cc2)=O)=O)CCC2(C1)CN(C(c1oc(C)cc1C)=O)C2 C1(C(N(CCCNC(CNS(CC)(=O)=O)=O)CC)=O)CN(C)CC1C(F)(F)F.C(CF)C CC(C)C(O)C(F)(F)C(=O)NCCCC(C)NC(c1csc(Cl)c1Cl)=O n1(CC)ccc(C(=O)NC2CC(C)C2)c1.c1(C2(C(=O)N)CC2)noc(C)n1 C1(C(=O)NCCN(CCCC)C)C=CCN(C(C2C(C)C2C)=O)C1 N1(C(C(=O)NCCc2nc(CC)on2)=O)CCN(C2CCCN(C)C2)CC1 C12(c3n(-c4ccc(C)cc4)nc(CO)n3)COC(CN1Cc1sccn1)C2.OC c1(NC)ncccc1C(=O)NCCCNC(c1cn(C)c(C)n1)=O.C12CC1OC2 N1(C(C=C=C(C)C)=O)C2CC1CN(C(c1coc(C(N)=O)c1)=O)C2 N1(C(c2c(CC)noc2)=O)CCC2CCN(C(c3c(O)ccc(Cl)c3F)=O)CC12 N1(CC(=O)Nc2cccc(-c3c[nH]c(=N)[nH]3)c2)C(=O)N2C3CCCC2(C3)C1=O c1(OC)cccc(C(C)C(=O)OC(C2CCN(c3nc(C(F)(F)F)ns3)C2)C)c1 CCC(C)(C)CCCC(=O)N1CC(C(=O)NCC(C)(O)C(=O)OC)OC(C)C1 c1(C(=O)NC2C(NC(Cc3c(O)ccc(C)c3)=O)C2)c(C)[nH]c2ccccc12 C(N=c1cc[nH]c(C#N)n1)C1CCN(C(c2n[nH]c(C)c2O)=O)C1 C12(NC(C(C)N3CCC3)=O)CC(C)(C1)OC21CN(C(c2ccc(Cl)o2)=O)C1 C1(C(=O)NC(c2nc(C)[nH]n2)C)CCCCN1C(c1csnn1)=O C(=O)(CCC(C)(F)F)NCCCCN(C)C(C1CC1C(C)(C)C)=O C1(=O)C(C)(CF)OC(=O)N1.n1(CC(C)(C)O)ccc(C(=O)OC(C)(C)C)n1 C12(CNC(c3cn(CCCF)nn3)=O)CC1CN(C(c1ncsc1C1CC1)=O)C2 C1(CN(C(=O)Cc2nc(=N)[nH][nH]2)C)COCCN1C(=O)CC1CCCOCC1 C12(NC(C3CCC(C)C3)=O)CC(C1)N(C(c1ccn(C)n1)=O)C2 c1(C(=O)NC2CCOCC2C(N2CC(F)C(F)C2)=O)ccc([N+](=O)[O-])[nH]1 CC(O)C(C)C(=O)N(CC(C)(C)CNC(=O)C(C)NC(=O)C(C)(C)C)C C(=O)(C1=CC2CCCC12)N(CCN1CCN(C(C(CSC)(C)C)=O)CC1)C c1(C(=O)OCC)nccc(NC(c2nnnn2C(C2CC2)C)C2CCC2)n1 N1(C(CCN(CC)CC)=O)CCC(F)(CNC(=O)CC(C)SC)CC1 C1(CNC(c2c(C)csc2)=O)CN(C(=O)CSc2ccncc2)CC1C c1(CC(CNC(c2ccccc2Br)C)=O)ccccc1F N1(C(C2C(CC)CCC2)=O)CCC2(C1)CN(C(c1c(OC)cccc1C)=O)C2 N1(C(c2csc(Cl)c2)=O)CCOC2(CCN(C(C3(CN(C)C)CCCC3)=O)C2)C1 c12csc(c1)C(=O)NC2.C(C(CO)n1cccn1)NC(C1C(C(C)(F)F)C1)=O CC1CCCCC1n1nc(-c2ccc(N)cc2)nc1-c1cc(Cl)no1 C1(NC(CC(C)(C)OC)=O)CCCCN(C(=O)C(C)(C)F)C1 c1(C(=O)NC(C(=O)N(CC)Cc2ncc(C)[nH]2)C)nn(C)cc1C CC#CCC(C(=O)NC1CCC(OC)C1)NC(c1ccc(CC)cc1)=O c1(C(N(C2CCCCC2)CC)=O)cc(CNC(c2ccc(C)[nH]2)=O)no1 CCCC(C(=O)NC1CCC(CC(N2CCC(CN(C)C)C2)=O)CC1)NC(N)=O CC(O)C(C(=O)N(CCCOCCN)C)N.C(=O)(C1=CSCS1)N(C(N)=O)C N1(C(C(C)(O)C2CC2)=O)CCC2(COC(CNC(c3cccc(=S)n3O)=O)C2)C1 CC(C)C(C)(CNC(=O)CC1CCC(=O)N1)NC(=O)CC1CSCCO1 C#Cc1ccc(Cl)c(C(=O)NCCC2(CNC(C3CC3(C)CC)=O)CC2)c1 C1(OCC(C)=O)CCN(C(C2(C3OCCC3C)CC2)=O)CC1 C1(NC(C=CC)=O)CN(C(c2ccn(C(C)(C)C)n2)=O)C2(CCC2)C1 NC(=O)CCCCC(=O)NC1CC(O)C1CC(=O)NC1(CC2CC2)CC1 c1(C(N2CCC(NC(c3c(C)cco3)=O)CC2C)=O)cnc(C)c(C#N)c1 CC(O)C(C(=O)NCC1CC(CO)CN1C(=O)CN(c1cccnn1)C)N(C)C C=CC(C)C(C)C(=O)N(CCCN(C)C)CCNC(c1c[nH]ccc1=O)=O C(=O)(CC1=CCN(C)CC1)N1CCC(C2(NC(c3ccc(C)c(F)c3)=O)CC2)C1 C1(C(C)(C)C(=O)N2CC(C(=O)Nc3cccc(C4CC4)c3)C2)CN2CCC1CC2 c1(NC(N2CCC(C)(CNC(=O)Cn3cc(CO)nn3)C2)=O)cc(F)ccc1F C1(N(C(C2CCC2(C)C)=O)CC)CCCN(C(c2ccc(C(C)F)cc2)=O)CC1 Cc1ccc(C)c(SCC(=O)NCCNC(=O)COCC2(F)CC2)n1 C(=O)(C1=CNC2=NCCCN12)NC1C(NC(CC(C)(C)C2CCCC2)=O)CCC1 CC1(C)OCc2c1n[nH]c2C(=O)NC1CCC(NC(C2CCOC2(C)C)=O)CC1 c1(C(N)=O)ccccc1C(C1CCCO1)NC(C1CCCN(C(=O)CC(N)=O)C1)=O N1(C(C2(CC)CC(C)(C)C2)=O)C(C(=O)NCCCN(C)C)C2CC(O)C1C2 C1(C(=O)NCCCOC(C)C)COC2(C1)CN(C(C1(C)CC3C=CC1C3)=O)C2 O=C(CCCCO)NCC(N1CCC(N(C(=O)C(O)C2CCCC2)CCO)C1)=O C1(NC(C2CC3CCCCC23)=O)CC2CC(NC(C3(C(F)(F)F)CCC3)=O)C1C2 N1(CC)CC(NC(=O)CC2CC3(C2)CN(C(C2(CC4CC4)CC2)=O)C3)CCC1=O C1(C(N2CCC(C(N(CCCC)CC)=O)(CF)C2)=O)C2CCC(C2)C1C N1(C(C(=O)NCC)=O)CC(C)CCC1CNC(=O)CCCNC(C)=O CCC(F)(F)C(=O)NCC1(C(=O)N(CC(C)C#N)C)CC(C)(C)C1 C(C1CCCN1C(=O)Cn1ccccc1=O)=CC(=O)NC1CCCOC1 CCC(C)C(C(=O)N1CC(CC(F)F)C1)N(C)C(c1ccc([N+](=O)[O-])o1)=O C(=O)(CCC(C)SC)NC(CC)CN(C(=O)C(C)=C(C)C)CC c1(C(N2CC3C(C(N4CCC(C(N)=O)C4)=O)C3C2)=O)ccnc(F)c1F c1(NC(C(C2CCC2)NC(C2C(OC)(OC)CC2)=O)=O)ccc(C2CC2)cc1C Cc1ccc2cc(C(=O)NCC3CCN(C(=O)CC(C)CF)C(C)C3)ccc2c1 N1(C(CN(CC)CC)=O)C2CCC1CC(O)(CNC(=O)Cc1csnn1)C2 N(C(=NCCc1cccs1)NC1CCN(C(=O)C(C)(C)C)CC1)CC(COC)F N1(C(COCC(C)(C)C)=O)CC(CNC(=O)C2=CCCOCC2)OC2(CCC2)C1 N1(S(=O)(=O)c2cnn(-c3ccccc3)c2)CCC2(CCCN2C2CCNC2=O)C1 C(=O)(C1CCc2nccn21)N1CCC(CCCNC(=O)CC2CCC(=O)N2)CC1 C(=O)(C1CCOc2ccccc21)N1CCC(NC(CCC(C)C)=O)C12CC2 CC(CC(=O)N1CCN(Cc2c[nH]c3cccnc23)C2CC12)CC(C)(C)C c1(CC)ocnc1C(=O)N(C1CCCC1)CCNC(C1CCOC1C(F)(F)F)=O C(=O)(C1CCCc2cncn21)N1CCCC(N(C(Cc2c(C)noc2C)=O)C)C1 C=CCC(C)(C)C(=O)NCC1CN(C)CCN1C(C1CCC(C2CC2)C1)=O C(=O)(C1=NOC2(CCOC2)C1)N(C)CCC1CCCCN1C(=O)C(C)(C)CO CON(CCCO)C(=O)C1(C=C)CCN(C(C2CCCCC2O)=O)C1 c1(C(=O)NCCC(C)NC(c2c(C(C)C)nns2)=O)ccc(N)c([N+](=O)[O-])c1 C1(C(C)NC(=O)Cc2nnc(O)s2)CN(C(c2ccc(Cl)o2)=O)CCO1 CCCCCCC(C)CC(=O)NCC1CCN1C(c1ccc(Cl)cc1)=O N1(C(C(C)CCO)=O)CCCC(C2CCN(C(=O)CCn3cccn3)C2)C1 Cc1nc2cc(C(=O)NC3CCCC3CNC(=O)Cn3cncc3C)[nH]c2s1 N(C(=NCCSC)N1CCC2(CCc3ccccc3O2)C1)C(CC)C C(=O)(CC(C)CC(C)(C)C)N1CCOCC(C(=O)N(C2(C#C)CCOC2)CC)C1 N1(C(C(C)CC2CCC2)=O)CCC2C(C(=O)NCC3CCCOC3)C2C1 C(CCC(C)(C)NC(=O)C(C)CC1CCCO1)NC(Cc1c(C)nc[nH]1)=O c1(C(=O)NC2(CO)CN(C(C(CC)C)=O)C2)cccc(Br)c1 C1(NC(CCOCCOC)=O)CN(C(c2cc(C3CC3)cs2)=O)C2CCCC12 C(=O)(CCC(CF)CF)NCCCN(C(C1C(C)(C(F)F)C1)=O)CCO Cc1nn(C)c(C(=O)NCCC2CCCN(C(C3CC3CF)=O)CC2)c1Cl Cc1cncc(C(N2CC(CNC(c3cc(CCO)on3)=O)CC(C)C2)=O)c1C c1(OC)ccc(C)c(-c2ccnc(CC(=O)NC(C)C#N)c2)c1 N1(C(C(CC)Oc2ccccc2)=O)CC(NC(=O)C(F)=C(C)C)CC(F)C1 CCC1=NOC(C(=O)NCC(C(=O)NCc2cscc2C)OC)C1 C(=O)(C1=CCN(C(=O)C(C)n2ccnc2)CC1)NCCN(C)CC Cc1cc(C(=O)NC2(CO)CCCN(C(C3COCCO3)=O)C2)cc(C)n1 C(C1C(C(=O)NC2(CCCNC(=O)C=C(C)c3cccs3)CC2)C1(C)C)=C(C)C C1(NC(C2=CC(C)(CC)C2)=O)CC2CCC1CN(C(=O)C(C)COC)C2 c1(CCNC(=O)NCc2cc(C#N)cc(Br)c2)cccc2cnccc12 c1(C(=O)NC2CC(CNC(=O)C=C3CCCCC3)C2)cc(F)cc(F)c1 N1(C(CCCSC)=O)CCOC2(CCN(C(=O)C(n3nccc3C)C)C2)C1 CC(C)CC(C(=O)NCC1CCN1C(C1(C)C=CCC1)=O)C(N)=O c1(S)ccc(Br)cc1F.c12nn(C)cc1-c1cn(nn1)CC1CCCN1C2=O.CO c1(C(=O)NCC(C)NC(c2cc(OC)no2)=O)cc(C)cc(F)c1N C1(NC(CN2CCN(C)CC2)=O)CCN(C(c2cccc(C#N)n2)=O)CC1(C)C Cc1cnccc1C(C)C(=O)N1CC(N(C)C(C2CCCCN2C)=O)C1 c1(CC(=O)N(C(C)CNC(=O)CC2CCCCO2)C)ccccc1Cl c1(C(=O)NC2(C(=O)NC3CC(C)(NC(CC4C(C)C4)=O)C3)CC2)ccccc1Cl C1(CC(=O)NCCC(C)CCNC(=O)C=CC2CCCCC2)(OC)CCOCC1 CCN=c1[nH]cc(C(=O)NC2CCC(C)N(C(c3cccc(OCC)n3)=O)C2)s1 C1(CNC(c2nc(C(C)NC(c3sccc3F)=O)oc2)=O)CCCNC1=O N1(C(Cc2nc(C)oc2)=O)CC2CCC1CN(C(=O)CC1(C(F)(F)F)CC1)C2 N1(C(Cn2nnc(=N)[nH]2)=O)CC(NC(=O)C=CC2CCC2)CC2(CC2)C1 c1(OC)cc(NC(C2CCC2CNC(=O)C(C)(O)C2CC2)=O)ccc1C C1(NC(c2[nH]cc(C(N)=O)c2)=O)CC(NC(c2csnn2)=O)C12CCC2 N1(C(C2(C)CCOC2)=O)CCN(C(=O)CC(C2CC2)C2CC2)C(C2CCC2)C1.CO CC1c2ccccc2OC1CC(N1CCC(N(C(=O)C(C)(C)C(F)F)C)CC1)=O C1(N(C(CCC)=O)C)CCCN(C(=O)CC(COC)c2ccc(Cl)cc2)C1 N1(C(c2c(CNC(CC3(C(=C)F)CCC3)=O)noc2)=O)CCSCCC1C CC(C)CC(C)(O)C(=O)N1CCCC(C(=O)NCCc2ncnn2C)C1 C1(CCC)CN(C(=O)Cn2ccc(C)c2)CCN1C(=O)C(C)c1cc[nH]n1 c1(COC)ccoc1C(N1CCCC1CCC(=O)NC(c1n[nH]c(C)n1)C)=O C1(C(=O)NCC(C)N(C)C(c2ncc(C3CC3)cc2F)=O)CC(=O)NC1(C)C N1(CC(C(C)C)O)CCCOC(CNC(c2scnc2Cl)=O)C1 C1(NC(COC(C)(C)C(F)(F)F)=O)CCCCCC1NC(C1(C)CC1(F)F)=O C1(C(=O)OCC)CN(C(C)=O)CCN(N2C(C=O)COC(=O)C2)C1.C(C)(C)C CC1CC(NC(C2CCCC(C)(C)C2)=O)CCN1C(C1(F)CCCC1)=O N1(C(C(C)SCC(C)C)=O)CC2C(NC(=O)C(CC)Sc3ccccc3)C2C1 c1(C(=O)NC2CCCC(NC(C(C)O)=O)C2)ccc2nc(O)oc2c1 c1(C(N2C(CN(C(C3C(CC)C3)=O)C)CCC2)=O)cc(Cl)c(Cl)cc1C N1(C(C2N(C)CCOC2)=O)CC2(C(=O)O)CCC2(C(=O)O)C1 c1(C(N2CCC(C(C(=O)N(CC(CC)CC)CCC)F)C2)=O)cnccc1C C1(C(=O)NC2(c3onc(C)n3)CC2)CCOCC1NC(C1(n2nccn2)CC1)=O C1(NC(CN2C(C)CCC2)=O)CC2CC(NC(=O)Cn3cnnc3)C1C2 C1(CC=C)(CNC(c2cc(OC)cs2)=O)CCN(C(=O)C(O)CCSC)C1 Cc1ccc2oc(C(=O)NC(C)(CNC(C3CCC3(C)C)=O)CO)cc2c1 c1(C(=O)NC2C(NC(C(CC)C)=O)CCCC2)nn2c(c1C)CCCC2 C(C)(C)(CCCCNC(=O)C(C)SC)NC(CCCCOC)=O CC1CCC=C1C(=O)NC1(c2ccccc2)CC(NC(C2CC(F)(F)C2)=O)C1 N1(C(CC=CC)=O)CC2CCCN(C(=O)CC3CCCC3O)C2C1 Cc1cc(F)ncc1C(=O)NCC1(CSc2ccc(O)c(Br)c2)CC1 c1(-c2ccc(C(=O)OC)nc2)cc(C(=O)OC2(C)CCOCC2)ccc1OC c1(NC(CCCC)C)ccc(S(=O)(=O)NCc2coc(C(C)(F)F)n2)cc1Cl C1(NC(C2C(=C)CC2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 c1(NC(=O)NC(COCCC(=O)OC)=O)ccc(SC)cc1OC(C)C.OC CC1(C)CC(NC(C2CCC(O)C2)=O)CN(C(C2(C(C)(F)F)CCC2)=O)C1 C1(=O)CC(O)CN1.C1(CN(C(=O)COCC=C)CC#C)CCCO1 C12(CNC(c3cnc(C)[nH]3)=O)CCCC1CCN2C(=O)CNS(N)(=O)=O C1(C(=O)NC2(COC)CN(C(=O)CCCCCc3cccs3)C2)CCN(C)S1(=O)=O c1(CCC(=O)NCC2CCN(C(=O)CC3CCC3(F)F)CC2)cccc(F)c1 C12(C(=O)NCC3CCN(C(c4nc(C)sc4)=O)CC3)CCCC1CS(=O)(=O)C2 N1(C(COCC(=C)C)=O)CCC(C2CC2)C1CNC(=O)C=CCN(C)CC C1(C(=O)NCCNC(=O)CSC(F)(F)F)CCc2ncncc2C1 N1(C(C(C2CC2)OC)=O)CC(NC(=O)CCCCC2CC2)C(Cl)C1 Cc1cc(C(N2CCOC(CNC(=O)CN3CC4CC4C3)C2)=O)nc(O)n1 CC(CC1CCC1)C(=O)NC1(C(=O)N(C2CCC2)C2CC2)CCCC1 N1(C(CCNC(CC(C)C)=O)=O)CCC(NC(c2ccc[n+]([O-])c2)=O)CC1C C#CC1(C(=O)NCCN2CCC(C)CC2)CCN(C(c2cn(C)cn2)=O)C1 C(=O)(CCC(C)C)NCC12CC(C(=O)Nc3n(CC)ncc3)(C1)C2 CCC(CC)(CCNC(c1nnn(C)c1C)=O)NC(=O)C=Cc1nccs1 Cc1noc2nc(C(=O)NC34CC(NC(C5C6COCC56)=O)(C3)C4)ccc12 N1(C(Cc2c(C)noc2C)=O)C2CCC1CC(NC(=O)C(C)P(C)(C)=O)C2 N1(C(C2(OC)CCC2)=O)CCC(NC(=O)C=Cc2cncc(C)c2)C2(CCC2)C1 c1(C(N2CCC(N(C)C(C34CCC3CC4)=O)C2)=O)cnc2ccoc2c1 N1(C(C=CCCC)=O)CC(CCNC(c2ccc(C(N)=O)nc2)=O)OC(C)C1 C(=O)(C(CNC(c1cccc(Cl)c1)=O)CC(C)C)NCc1ccc(C)c(F)c1 Cc1oc(C)c(C(=O)NCC(C)(O)CNC(=O)C(F)C(F)(F)F)c1Br N1(C(C(=O)NCc2ccc(OC)cc2)CC2(C)CCOC2)CCC(S(N)(=O)=O)C1 CC1OC2(C)CC1(C(N1CC(NC(C34CC(C)(CO3)C4)=O)C(F)C1)=O)C2 C1(CN(C(=O)C(C)N(C)C(C(C)(C)CC)=O)CC)CC(F)(F)C1 C1(C(=O)NCCCOCCNC(Cn2ccc(C)c2)=O)COCC(C)O1 Cc1cc(-n2nc(CCCN(C)C)nc2-c2cc(O)ncc2Br)cc(F)c1 C1(C(=O)NCCN(CCC)C(c2nnn(C)n2)=O)CC(c2cccc(F)c2)=NO1 C1(NC(C2C(NC(C(CC)n3ccnc3)=O)CCO2)=O)CCN(C)CC1(C)C c1(C(N2CCCC(CCC)(NC(CCC)=O)C2)=O)ccc(Cl)c(Cl)c1N c1(C(C(=O)NCC2(CNC(C3CC(N(C)CC)C3)=O)CC2)C)ccnn1C N1(C(c2c(C)cc(CNC(CC(CC)O)=O)o2)=O)CCC2(CCCCO2)C1 CCCCCCCCC(=O)N1Cc2[nH]nc(C(N3CCOC(CC)C3)=O)c2C1 C#Cc1ccc(C(=O)N(CC(N2CCOC(CC)CC2)=O)C2CC2)cn1 C1(CNC(C(C)OC)=O)CN(C(c2csc(SC)n2)=O)CCC12CCOCC2 CCCC(CCNC(C12CC(CO1)N(C(c1nc(C)ccc1C)=O)C2)=O)CCC c1(C(=O)NC(CNC(COC)=O)C(C)(C)C)cnc(C)[nH]c1=N c1(CC(=O)NCCCCN(C(=O)CCCc2ccncc2)C)ccsc1Cl C1(N(C)C(c2ccc3nnn(O)c3c2)=O)CCc2[nH]c(=N)sc2C1 N1(C(c2ncc(C)nc2)=O)CCC(C(=O)NCC2CCC2C)C(C)C1 C(=O)(C(C)(O)C(C)C)NCC(CCNC(c1cn(CC=C)nn1)=O)(C)C c1(N(C)CC2CCCN2C(c2cc(Cl)nc(Cl)c2)=O)nc(O)c2c[nH]nc2n1 CC1(C#CC(=O)N2CCC(CF)(NC(C3CC3C(F)F)=O)C2)CCCO1 C12(CNCC)COC(C1)C(O)C2.C1(=O)C(C)(O)CCCOc2cccc(c2)CO1 C=CC1(CC(=O)NC2CN(C(c3csc(C(C)C)n3)=O)CCC2C)CCOCC1 CCCC(CC)CC(=O)NC(CC)(CC)CCNC(=O)CN1OC(C)(C)CC1=O CC1(C)c2ccccc2CN1CCS(=O)(=O)c1ccccc1Br CC(C)S(=O)(=O)CC(=O)NC1(C2CCCN2C(=O)Cc2ccnc(Cl)c2F)CC1 n1(CCCC)nnnc1C(C)(CCCl)NCC(F)C(=O)OCC C1(CNC(COC)=O)CCN(C(=O)CCOCC(N2CCOCC2)C2CC2)CC1 N1(C(C2(C(C)(C)O)CC2)=O)CCC(NC(c2sccc2Cl)=O)C(CO)CC1 C(=O)(C1CCOc2ccc(Cl)cc21)N1CC(CNC(COCCOC)=O)OCC1 C1(CN(C(=O)C2=NOCC2)C)CCCCN1C(C1CCCN1C=O)=O c1(NCCNC(C2CCCCN2C(=O)C=CBr)=O)ncc2ccnc-2[nH]1 CCC(CSc1ccccc1)CC(=O)N(C)CCNC(C12CC(F)(C1)C2)=O c1(OCC)ccccc1C(N1CC(F)(CNC(=O)CC2CCCSC2)C1)=O C1(CC)(NC(c2nocc2Cl)=O)CCCN(C(=O)Cc2ccnc(O)c2)C1 C(=O)(C(CC)C(=O)N(C(C)C(=O)NCC1(C(O)COC)CC1)C)OCC c1(OC)cnnc(C(N2CC(C)(OCC(=O)NC)C2)=O)c1.C1COC(C)C1 N1(C(CC(=O)N(C)C)=O)C2CCC1CN(C(C1CN3CCC1CC3)=O)C2 N1(C(c2cccc(C(C)O)n2)=O)CCCCC(C2CN(C(=O)C(C)C)C2)C1 C1(C(N2CC(CC)C(C(=O)NC(C)C(C)(C)C)C2)=O)CC2(CC2)CN1C N1(C(CCC2OCC(C)(C)C2)=O)CC2(CCC(CNC(=O)CC3CCC3)O2)C1 C1(O)CCS(=O)(=O)C1.C(C1CCCC1)=C(C(=O)N)C.C1C(=O)NCCOCCOCC1.CC=C C1(NC(CC2N(C)CC=CC2)=O)C2CCC1N(C(=O)Cc1ccon1)C2 C1(=O)C2=CCN(CC2)C(=O)C2(CCC(C)C2)N1.c1(C(CC)CC)cccs1 C1(NC(C2(C)CCCS2)=O)CCN(C(c2ccsn2)=O)CC1CO C1(N(C)C(C2CC(OC(F)F)C2)=O)CCCCN(C(=O)C(F)(F)C2CC2)C1 C12(NC(C(C(C)C)OC(C)=O)=O)CCC(C(=O)NCC3CCOC(C)C3)(CC1)C2 C#CCCCC(=O)NC1CC2(C1)CC2NC(c1c[nH]cc1Br)=O CC1=NOC(=O)CN1C(=O)Nc1ccc(N2CCOCC2=O)nc1 N1(C(C2N(C)CCOC2)=O)CCC(CNC(C2CC3CCC2O3)=O)C(F)(F)CC1 C(CN=c1ncc(O)c[nH]1)C1N(C(c2c(C)nn(C3CCC3)c2)=O)CCCC1C C1(CNC(C(C)C=Cc2ccccc2)=O)CC(F)(F)CN1C(=O)Cc1cocn1 O=S(=O)(c1ccc(OC)c(Cl)c1Cl)N(CCCO)Cc1nccs1 C1(NC(C(C)OCC#C)=O)CC12CCN(C(=O)Cc1cccs1)CC2 C1(NC(=O)COC2(CCCCN(C(CC=C)=O)C)CC2)CCCOC1C C(=O)(C(C)(C)CCCNC(=O)CCC1CC1)N1CCC(C)C(CO)C1 C1(CNC(C2(OC)CC2)=O)CN(C(=O)C(CC(C)C)NC(C)=O)CCC12CCC2 C123CCC(CC1)(C2)n1cc(nn1)CCC(=O)N3CCO.C1(C(=O)O)CC12CC(O)C2 c1(CC(=O)NCC2CCCCO2)c(F)cncc1Cl.c12cn(nn1)C1CN(C1)C2 C1(N(C(C(C)CO)=O)C)CCN(C(=O)Cc2ccccc2)CC1.C(S(C)(=O)=O)CC Cc1sc(O)nc1C(=O)NCC(C)C(=O)NCC(n1ccnn1)C c1(OC)cc(C(=O)NCC(C)(C)CCNC(=O)CC(=O)NC2CC2)ccc1F N1(C(CNC(CC)=O)=O)CC2CN(C(C3CC34CCCCCC4)=O)CC2C1 c1(NC(Cc2ncc(COC)s2)=O)cccc(CN2CCCNC2=O)c1 N1(C(c2ccc(SC)o2)=O)CCN(C)CC1CNC(c1ncsc1C)=O Cc1c(CNC(=O)NC2(CCF)CCOCC2)cccc1F C(=O)(CCCCCCNC(=O)C(=O)NCC12COCCN1C(=O)COC2)OC C1(C2CN(C(c3nnc(Cl)cc3N)=O)C2)(NC(CC2N(CC)C(=O)CC2)=O)CC1 Cn1cc(-c2ccccc2)cc1C(N1CC=CC(NC(=O)C(O)C2CC2)C1)=O C1(NC(C(COCC)(C)C)=O)CC2CCC(C1)N2C(C1CC(CC(=O)OC)C1)=O Cc1ccc(CC(=O)N(CCC(C)N(C(C2(c3ccsc3)CC2)=O)C2CC2)CC)s1 c1(C(=O)NC2CC(C(=O)NCCCOC)C2)nnc(S)n1C c1(C(N2CC(C)(NC(c3cccc(OC)c3O)=O)C2)=O)cc(Cl)cc(F)c1F C1(C2CC2)(CNC(CCC(C)(C)C)=O)CCN(C(=O)CC2CCCNC(=O)C2)C1 c1(NC(C(C2CCOC2)OC)=O)cccc(CSN2CCCCC2)c1 N12CCCC1C2=O.N1(CC)CCC1CC(=O)NC12CC(C1)C2 C1(OCC)COCCC1CC(=O)N(C)CCNC(=O)C=C1CCCCC1 c1(NC(=O)C(c2ccccc2)O)ccc2[nH]c(C(=O)N=c3cco[nH]3)cc2c1 N1(C(C(C)CF)=O)CCN(C(=O)C2=CCCCC2)CC12CCC2 C1(NC(C2N(C(C3CCCC(=O)C3)=O)CCC(=C)C2)=O)CCc2ncnn2C1 c1(NC(=O)NCCOC(CN(CCC)Cc2ccco2)=O)cc2ccccc2o1 N1(C(C=CC=CC)=O)CCC(C2CC2)C1CNC(=O)COC1(C#N)CCC1 CC1CC(NC(=O)C(C)(C)c2cnsc2)CCN1C(c1cc(Cl)c(Cl)[nH]1)=O c1(C(=O)OCC)cc(S(=O)(=O)Nc2ncc(OC)c(C)n2)cn1C C1(C)(NC(c2nc(CC)sc2Br)=O)CCN(CC#N)CC1 Cc1cc(C)c(C(=O)NC(CCN(C(=O)C(C)CS(C)(=O)=O)C)C(C)C)c(=O)o1 CCC(C)(CCC(C)C)C(=O)NCC1CN(C(=O)CC2CCOCC2)CCCO1 C(=O)(C(C)N(C(=O)CCOCC)C)N(CC(=O)NC)CC#C.N(CC)CC c1(C(N2C(CC(=O)Nc3c(C(=O)OC)n[nH]c3)CC2)=O)cc(C)[nH]c1C c1(C(=O)NCc2c(C(=O)NCC3(CCC)CCC3)cco2)cc2ccccn2c1 N1(C(=O)NC2CCC(Cc3ncoc3Br)C2)CCC(F)CC1 c1(CC(=O)N(CCC)CCNC(=O)CCC(C)(F)F)ncn2c1COCC2 Nc1ccnc2c(C(N3CCCC3CNC(c3ccnnc3O)=O)=O)cnn12 C1(CC(=O)NC(CNC(COC)=O)(C)C)CCC(NC(=O)Cc2ccccc2)C1 c1(C(=O)NCC(CCNC(CC(CN(C)C)O)=O)O)cnc2n1CCS2 CON(CCCO)C(=O)c1cc(CNC(=O)CCOC2CCC2)no1 C1(C(C)C(N2CCC(N3CCOC3=O)C2)=O)CCN(C(=O)Cc2ccco2)CC1 C1(CNC(C(C(C)(C)O)F)=O)CC12CCN(C(=O)C=Cc1cnccn1)CC2 c1(SCC(=O)NC(CNC(C2N(S(C)(=O)=O)CC2)=O)C2CC2)nnc(S)s1 c1(C(=O)NCC(CC(C)C)NC(c2c(C)n(C)nc2)=O)cc2ccc(O)cc2[nH]1 c1(CC(N2CCC(Cn3cc(CCN(C)C)nn3)C2)=O)csc2ccccc12 C(CC(F)F)(C(=O)N1CC(C)C1(C)C)N(C(C(C)Cn1cccn1)=O)C c1(C(N2CC(C)(C(=O)NCCCCCO)C2)=O)cc(Cl)cnc1F CN1N=C(C(=O)NCC2CCN2C(C2CCC=CO2)=O)CCC1=O c1(C(=O)NCCCOCCNC(C(C)CC2CCC2)=O)cn(C)c(=O)n1C c1(C(N2C(CN(C(C(F)=CCC)=O)CC)CCC2)=O)cc(N)c(Cl)cn1 C1(C2CCCC2)(C(N(C(CCNC(CN(C(=O)OC)C)=O)C)C)=O)CCNC1=O Cc1coc(C=CC(=O)NC(C)CCCNC(=O)CC2CCN(C)CC2)n1 C1(NC(C(CCC)NC(=O)COCCCN(C)C)=O)CCC(=O)NC1(C)C c1(Cn2cc(CN)nn2)cccc(CO)c1.C1(C(N2C(C)CC2)=O)CCOCC1O c12ncccc1C(=O)N1CC(C1)OC2.C1(C)(NC(CSCCC)=O)CC1(C)C C(=O)(C1CCCc2ncnn21)NC1CN(C(c2c(Cl)cc(C)s2)=O)CC1O C1(CN(C(C2(SC)CCC2)=O)C)CCCCN1C(C1CC(C)(C)O1)=O c1(C(N2CCN(C(C=Cc3c(C)ccnc3)=O)C(C)C2)=O)nc(O)nc(O)c1N N1(Cc2ccc(C)nc2)CCCN(C(=O)C(c2ccc(Cl)cc2)C2CC2)CC1C c1(C2OCCC2c2nc(C3(c4cncc(C)c4)CC3)no2)cc(F)cc(F)c1 c1(CC)c(C(=O)NCC(CCNC(c2ccon2)=O)OC)cccc1C C12(C(=O)NCCC(C)(C)NC(COCC(=O)NC)=O)CCCN(CC1)S2(=O)=O C#CC1CC2(CC(C(=O)N(C3CCN(C(C4CC4(F)Cl)=O)CC3)CCC)C2)C1 CC1SCCCC1C(=O)NC(C(=O)NCCN1CC=CC1)c1ccco1 C(c1cccnc1)=CC(=O)NCC1CCC(NC(C2CCC(O)N2)=O)C1 N1(C(C2N(C(c3cccc(C)c3F)=O)C(C)C2)=O)CC(C)CC(C)(C)C1 Cc1cccc2c1OCC2C(=O)NCC1(O)CCCN(C(=O)C2=NNC(=O)C2)C1 c1(OC)ccnc(OC)c1C(=O)NC1CCCCC1NC(=O)Cn1nccc1C C(=O)(C(C)(C)C(C)(C)O)NCC(CC)(C)C(=O)N(CCC1=CCCCC1)CCO n1(CC(=O)OC)cnc(C)c1C(=O)NC1COCC1NC(C1C(C)C1C)=O CCCCCC(=O)NC1C=CCN(C(C2(NC(C)=O)CCCCC2)=O)C1 N1(c2ncc(C)c(C)n2)CCC2C(CCCN2C(=O)C=Cc2cc[nH]n2)C1 N1(C(C(CCOCC)NC(c2cnc(C)cn2)=O)=O)CC(=O)NC(C)C1 C1(CNC(C(C)SCC)=O)CN(C(=O)CC(c2ccccc2C)C)CCC1C C1(C(=O)NCCCOCCN(C(C2CCC(CC)CC2)=O)C)CC12CCOCC2 Cc1ccc(C(N2CCC2CNC(C2CCC(C)(C)O2)=O)=O)cc1F c1(OC)ccc(C)nc1CNC(c1ccc(NC2CC2)nc1)=O CCCC(C(O)C(=O)N1CCC(CCF)CC1)NC(=O)CC(C)(C)C#N c1(CC)cc(=NCCC(C)NC(c2c[nH]nc2C(C)(C)C)=O)[nH]c(C)n1 n1(CCC)cc(Cl)c(C(=O)NCC(C)CNC(=O)Cc2cnnn2C)n1 c1(C(=O)NC2(CNC(C(CC#C)C)=O)CC2)ccc2cccnc2c1N N1(C(C(CC)OC)=O)CCC2CCCC(C1)N2C(=O)C(F)(F)CC(C)C C(C(C)(C)CC(=O)NC(c1cccc(C)c1)CNC(=O)C(O)CF)OC N1(C(N(C(C)C)CC)=O)CCCC(OCC(F)(F)F)C1 CCCCCN(CCC(=O)NCC(C)N(C(=O)CCNC(N)=O)CC)C N1(C(c2scc(OC)c2)=O)CCC=CC1C(=O)NCC(c1ccncc1)O C(=O)(C(O)CCCc1ccccc1)NC1CCN(C(C2CCC(=O)NC2)=O)CC1 c1(CC(=O)NCC#CCNC(C(c2cnn(C)c2)SC)=O)cc(F)cc(Cl)c1 C1(C)(C(N2CC(CNC(C3NC(=O)CC(C)C3)=O)C2)=O)CCCNS1(=O)=O C(=O)(C(CC)CC(C)C)N1CCC(CC(C)NC(CC(C=C)(C)C)=O)CC1 c1(C(=O)NC2CCC(NC(C(C3CCC(=O)CC3)F)=O)CC2)ncc(F)cc1F C1(CNC(=O)CCOC2CC2)CC2CCCC2N1C(C12CCCCC1OCC2)=O CC1(CN(C=O)Cc2nocc2Oc2ccccc2)CCCC1 c1(CC(N2CC(C)CC(NC(CC=C)=O)C2)=O)c[nH]c2c(F)cccc12 N1(C(=O)NCCN(CCOC)C)CCCCCC1c1ccc(C(=O)OC)o1 N1(C(=O)NCc2occ(C(N)=O)c2)CCOC2(CC1)CCS(=O)(=O)C2 CC1CC=C(C(=O)NC2CCCC2CNC(=O)C2=COCCC2)CC1 Cc1nc2n(c1C(N1CCOc3c(Cl)cccc31)=O)CC(C)(C)CC2 n1(CC)ncc(C(N2CC(CCCCNC(=O)CCCn3ccnc3)C2)=O)c1C N1(C(c2cnc(CC)nc2O)=O)CCN(C(C2(OC(C)C)CCC2)=O)C(C)C1 c1(C(N2CC(C)(NC(C3C(N(C)C)CC3)=O)C2)=O)ccc(P(C)(C)=O)cc1 C1(N(C)C(c2cc(Br)ncc2Cl)=O)CCc2ncccc2C1 C(N=c1[nH]c(=NC2CCC3CCCC23)c2[nH]ccc2[nH]1)c1ccc([N+](=O)[O-])cc1 c1(OC)ccc(NC(=O)C(c2cccc(Cl)c2)N(CC(C)C)C)c(OC)c1 Cc1nsc(Br)c1C(=O)N(CCCCCNC(c1c[nH]nc1C(F)F)=O)C C1(C(=O)NC(COC)CC(=O)NC(C23CCC(CO2)C3)C)CC2(CCO1)CC2 Cc1cc2nc(Cl)[nH]c(=NC3CC4CN(C(c5ccc(CO)cc5)=O)C4C3)c2s1 C=CCCCCC(=O)NCC1(CNC(C2CC2Cl)=O)CCC1 CC1CC(c2ccccc2)N(C(=O)NC2COCC(C)O2)CC1C C1(CC(=O)NC2CC(F)(CNC(C3CCC(=O)N3C3CC3)=O)C2)CCCOCC1 N1(C(C2(F)CN(C(C3CCC(CCCC)CC3)=O)C2)=O)CCCCC(C)(F)C1 C(=O)(N=c1cccn[nH]1)c1ccc(-c2ccc(SC)cc2Cl)cn1 c1(CCC)cc(C(=O)NCCOC2CN(C(c3cscc3OC)=O)C2)c(C)o1 C1(N(CC(=O)N(CCC#N)CCC#N)C)CCCC(C)(C)C1 N1(C(c2c(OC)c(Cl)ccc2)=O)CC2C(NC(=O)CC(C)(C)O)CS(=O)(=O)C2C1 CCCCCC(O)C(C)C(=O)NCCCC1(NC(=O)COC)CC1 C1(CNC(c2cc(OC)no2)=O)C2CCC1CN(C(C1CCC1(F)F)=O)C2 C1(NC(=O)NC(C(C)(C)CO)c2ccc(Cl)cc2)COCCC1(F)F N1(C(c2c(C#C)cnn2C)=O)CC2CCCC2(NC(c2cccc[n+]2[O-])=O)C1 Cc1nsc(NC(=O)NCCC(O)CNC(=O)OCC)c1Br.C(C)(C)(C)O Cc1cc(=NCC2CC3CCC(C2)N3C(=O)COc2ccncc2F)[nH]cn1 c1(CC(=O)NCC(CNC(c2cn(CCC)nn2)=O)OC)ccc(C(N)=O)cc1 N1(C(C2(C)CS(=O)(=O)C2)=O)CC(CNC(C2CCCNC2=O)=O)C(F)(CO)C1 C1(C(=O)NCC2CCN(C(c3c(COC)scc3)=O)CC2)CC2CCCC(C1)C2 c1(C(=O)NC(CCN(C(CCOCC#C)=O)C)C)ccc(S(N)(=O)=O)nc1 c1(CC(=O)NCC(C)CN(C)C(c2ncccc2F)=O)cccc2nsnc12 CC1=NC(C(=O)NCCC2CCN2C(=O)OC(C)(C)C)CS1 C=C(Br)CC(C)(C)C(=O)N1CCC(O)(CNC(C2(C)CC2(C)C)=O)CC1 c1(C(=O)NC(CC)(CNC(C2(F)CCOC2)=O)CC)c[nH]c2cc(Cl)ccc12 CC(=O)CCCC(C)C(=O)N1CCSCC1C(N1CCC(C)(N(C)C)C1)=O N1(C(CC2CN(C)C2)=O)CC(CNC(C2CCC(NC(N)=O)CC2)=O)CC1(C)C C1(CC(=O)N(C(C(=O)OC)C)C)CCC(NC(=O)C(C)N=[N+]=[N-])CC1 CON=C(C(=O)NC1(C)CCN(C(=O)Cc2ncccc2C)CC1)c1ccco1 C(=O)(C(N)C1(CC)CCC1)NCC=CC=C c1(C(N2CC(NC(C34CCOCC3C4)=O)C2)=O)ccccc1CO c1(C(N2CC(NC(=O)COc3ccsn3)CC(C)C2)=O)cccc2nnn(C)c12 N1(c2nc(C)nc(Cl)c2)CC2CCC(NC(=O)COC(C)C)CC2C1 C(=O)(CC(CN(C)C)C(F)F)N(CCNC(=O)CN1C(=O)C(=O)N(C)C1=O)CC c1(C(=O)NC(c2cn(C(C)C(C)O)nn2)CCC)conc1C1CCC1 C(CN=[N+]=[N-])(C(=O)NC(COC)C1CC1)NC(C1CCN(CC)C1)=O C12(CCN(C)CCOC)CCCN1C2=O.c1(C=O)cc[nH]n1.CO N1(C(C(COC)O)=O)CCOC2(CCN(C(=O)C=Cc3ccc(Cl)cc3Cl)C2)C1 C(CCCCC(=O)N1CCN(C(C2CCC(=O)O2)=O)CC1C1CCCC1)OCC C(=O)(C(C)(C)CC(=O)NC(C1CCCC1)CNC(C1CCCC(C)C1)=O)OCC c1(CCNC(C23CC(C(F)(F)F)(C2)C3)=O)ccnc(Cl)c1F N1(C(C2C(C(=O)Nc3ncccc3-c3cccc(F)c3)C2)=O)CC(F)(F)C(F)(F)C1 Cc1nc(-c2ccc(CN3CCOCC3)s2)sc1CN(C)C N1(C(c2ccc(N(C)C)nc2)=O)CCCC1C1CCCCN1C(=O)CCCC#N C(=O)(C(O)CCNC(n1cccnc1=O)=O)N(C1CCN(C)C1)CC Cn1cnc2sc(C(=O)NC34CC(NC(C5CCOCC5(C)C)=O)(C3)C4)cc12 C(CC(C(=O)NC1CCCCC1CC)NC(c1cc(OC)ns1)=O)OCC c1(OC)cc(C(=O)NC2(C(=O)NCC3CC3c3ccoc3)CC(O)C2)on1 C1(C(=O)NCC(C)S(N)(=O)=O)CCC2(CC2)N1C(C1CC2(CCC2=O)C1)=O C1(CNC(C2CC(NCCN3CCOCC3)C2)=O)CCCCNC1=O c1(NS(CCNC(=O)NC2CC2)(=O)=O)ccccc1-c1cn(CC2CC2)nn1 C1(C(N2CC(NC(c3n[nH]c(C)c3O)=O)C(C)CC2)=O)CC2CCCC(C1)C2 n1(C(C)C)c(C(=O)NC2CCC2NC(=O)CN2CCOCC2)cc2ccccc12 c1(-c2cc(C(N(C)CC3CN(C(C4N=C(C)SC4)=O)C3)=O)on2)cccc(C)c1 C1(C(=O)NCC(CN(C(=O)CN2CCCC2)C)O)CSCCS1 CC(C)CC(F)C(=O)N1CCC(O)(CCCNC(=O)CCc2cnn(C)c2)C1 C=C(C)CCCC(=O)NCCC(O)C(=O)NCc1nncn1C1CC1 N1(C(CCOCC(C)C)=O)CC2(COC(CNC(=O)C(=O)Nc3ncc[nH]3)C2)C1 C1(CC(c2n(C)nnn2)Nc2ccc(-c3nc(CO)no3)nc2)CCOC(C)(C)C1 c1(C(=O)NC2CCCC2CNC(c2ccns2)=O)ccc(O)c(C(N)=O)c1 C1(CC)C(NC(c2nc(Cl)oc2C)=O)CCCN1C(=O)C1=CCCC1 c1(-c2n(CCC)nc(-c3cccc(C(F)(F)F)c3)n2)csc2cc(C)ccc12 c1(CC)nonc1C(=O)N(CC(C)NC(c1cccn1C1CC1)=O)C C(=O)(C1=C(Cl)CCC1)NCCC(C)N(C)C(C1CC(CC2CC2)C1)=O O=C(CCCn1cccn1)N1CC(NC(c2ccccc2)=O)C1C(F)(F)F c1(CN(C)CC2CCCN(c3ncc(I)cn3)C2)ccc(Cl)cc1Cl N1(C(CC=CC=C)=O)CCC(CF)(NC(=O)C2CC2)C1 C(=O)(C1=C(C)CCCC1(C)C)N1CC(NC(CCC(CC)C)=O)(CO)C1 C1(C(=O)NCc2n(C)ccn2)CC(=O)N(C2CN(C(C3CC(=O)N(O)C3)=O)C2)C1 C1(NC(C(C=C)O)=O)COC2C(NC(c3csc(C(C)OC)n3)=O)COC12 C12(NC(CS(C)(=O)=O)=O)CCC(CC1)N(C(c1csc3cccnc13)=O)C2 CC1(C(=O)NCC23CCCCC2C3)CCN(C(C23CCC(CC2)C3)=O)C1 c1(C(=O)NCC2CN(C(C(COC)C)=O)CC2C)ccc([N+](=O)[O-])c(C)c1 C1(C(CNC(C2C(CCC)CCC2)=O)O)CCN(C(C2CCO2)=O)CC1 c1(C(=O)NC2C(C)CN(C(=O)CCc3ccon3)C2)cc2n(c1)CCCC2 c1(CNC(C(CSCc2ccc(CC)cc2)C)=O)cc(OC)ccc1Cl S(=O)(=O)(c1cnc(NC2CCC2C)c(Cl)c1)N1CC(CC)N(C)CC1 C(=O)(CC(COC)NC(c1nnn(C)c1N)=O)NC(c1n(CC)ccn1)C c1(CC)c(NC(c2ccc(C3(OC)COC3)cc2)=O)cnn1CC c1(C(=O)NC)ncccc1Br.C1(CNC(CN(CCC)C)=O)COC(CN)C1 C(=O)(CS(=O)CC)N(C(C)C(=O)N(C(C)C(F)F)C)CCC c1(CC)nc(C)c(C(C)NC(C2CN(C(=O)CCC3CCCOC3)C2)=O)s1 CC(C)(C)CC(=O)N1CC(O)(CCNC(C2CCC(C(N)=O)C2)=O)C1 CCCCC(C)CCC(=O)N(CC(C)N(C)C(c1ccc(C)nc1C)=O)C C(CCC(C)C(=O)N1CCC(CNC(=O)Cc2ccco2)C1)OC N1(CCC(N2CCC(CNC(C3(C=C)CCC3)=O)C2)=O)CCN(CC)CC1 C1(N(C)C)CC12CCN(C(C1N(S(CC)(=O)=O)CC(N(C)C)C1)=O)CC2 N(C(=NC1CCS(=O)(=O)C1)NC1CCS(=O)(=O)C1)Cc1ccc2c(c1)N(C)CC2 c1(C(=O)NC2C(NC(=O)CC3CC4(CC4)CO3)CCCC2)cc2ncccc2[nH]1 N1(C(C2(C)CC2(F)F)=O)CCN(S(=O)(=O)c2cn[nH]c2)C2(CC2)C1 C1(CC)CCCC1C(N1CC(CN(C)C(c2nocc2C)=O)C1)=O Nc1cc(Cl)ccc1C(=O)NCC1(NC(C2CSCCS2)=O)CCCCC1 c1(C(=O)NC2CCC(CC(=O)NCc3c(C)nsc3)C2)cccc2c1CCC2 C(=O)(C1=Cc2ccccc2OC1)NC(c1ccc(SC(F)(F)F)cc1)C CC(C)C(C(=O)NCC(C(C)(C)C)NC(=O)Cc1nccs1)C1CCC1 c1(CN(C)Cc2cccc(-c3nnn(C)n3)c2)cc(Cl)ncc1Br C(=O)(C(C)(C)CC(C)(C)C)N(C)CC1CCN(C(Cc2c(C)occ2)=O)C1 c1(C(=O)NC(C2CCN(C(CCCSC)=O)C2)(C)C)[nH]c2c(c1C)CCCC2 CC(C)(C#N)CCC(=O)N1CC2CCC1CN2C(=O)Cc1cc(C2CC2)no1 C#CCC(O)C(=O)N1CCC(OCCNC(=O)CC2CC(CF)C2)C1 C(C)(C(=O)NC(CO)C(C)NC(=O)CCN1CCCCC1)(C(C)C)NC(C)=O c1(CNC(C(CSCC)NC(=O)C=CC2(C)COC2)=O)cc(=O)cc[nH]1 CC12CCCC1N(C(C1CCCOCC1)=O)CCN(C(C1CCCCO1)=O)C2 c1(C(=O)NCC2C(C(N(C3CCCCC3)C)=O)C2)ccnc(O)c1F C(=O)(CCN1C(=O)COc2ccccc21)NC(C)CN(C)C(c1cnn[nH]1)=O c1(C(=O)OC)ccn(CC(=O)NCC2(NC(C3CC=CCC3)=O)CCOC2)n1 c1(C(N2C(COc3cccc(C)c3)CCCCC2)=O)cc(Cl)c(Cl)cc1N C1(C(N2CCCC(CNC(C(C(=O)OC)C)=O)CC2)=O)CN2CCCN1CC2 c1(CC(=O)Nc2cccc(CNC(C3C(C)N(C)CC3)=O)c2)cccc(F)c1F C1(CNC(CCC2(C)CC2)=O)CCSC12CN(c1nc3ccccc3s1)C2 C(=O)(C1=CC(O)C(NC(=O)C=C2CCC(C)CC2)C1)NCCC=CCC c1(C(=O)NC2C(CNC(c3nc(SC)sc3)=O)CCC2)ccc(C)nc1N O=C(C1CCCn2cnnc21)Nc1cccc(NC(c2cnns2)=O)c1 c1(-c2c(NC(C)=O)cccc2F)cc(O)cc2ccccc12 Cc1cnc2cccc(C(N3CC(NC(c4csc(-c5ncc[nH]5)n4)=O)C3)=O)n12 C1(NC(C2C(C)C2)=O)CN(C(=O)C(C)(C)Oc2ccccc2)CC2(CC2)C1 n1(CC)nc(C)c(CC(=O)NC2CCC(NC(=O)C(O)CC(F)F)CC2)c1C C(=O)(CC(C)(C)CCC)NCCN(C(C(CC#C)OC)=O)CCCN(C)C c1(C(N2CC(CNC(Cc3nc(C)oc3)=O)C3(C2)CC3)=O)cc2ccccc2[nH]1 CN1C(=O)C(NC(=O)C(N2CCCC(C)(CN)C2)=O)c2ccccc21 CN1CCC(C(=O)N(CCCN(C)C(C2C3CCCOC23)=O)C)CC1=O O=C1CC(c2cnn(C3CC3)c2)NC(=O)N1CC1CC1C1CCOCC1 N1(Cc2cn(C(C)C)nc2)CCc2c(CNCCc3ccccc3)n[nH]c2C1 c1(NCC)cccnc1C(N1CCC(N(C)C(c2c(C3CC3)noc2C)=O)C1)=O CCC(CC)C(C)C(=O)NC(CO)CCCCNC(=O)CCCOC(C)(C)C N1(C(c2ccc(N)cc2O)=O)CCC2(CCN(C(C3(N4CCCC4)CC3)=O)C2)C1 C(=O)(C(CC(C)C)c1ccccc1)NCCCCCN(C(C1CC(OC)C1)=O)C C1(CC(=O)NC2C(CNC(c3c(C)nn[nH]3)=O)CCCC2)CC2(CCC2)CO1 Cc1c(NC(=O)OC(C2(C(=O)C3CC3)CC2)=O)cccc1CC1(N)CCCCC1 n1(CC)nccc1CN(CC(O)CO)CCc1csc(-c2ccccc2)n1.SCC C1(NC(Cc2c(C)cccc2)=O)CCN(c2ccncc2)CC1(C)C N1(C(C2N(C)CC(F)C2)=O)CC2=C(C1)CN(C(C1CC3C=CC1C3)=O)C2 Cc1csc(=NCC(=O)N(C(C)CCNC(c2nnn(C)c2C)=O)C)[nH]1 C(C)(CC(C)(C)OC)NC(CN(C(C1C(CC)CCO1)=O)CC1CC1)=O C1(NC(C(CC2CC2)NC(=O)CCOC2CCC2)=O)CCCCCC1F CC(C)C(O)(C(=O)NC(C)CCNC(C1CCOCC1)=O)C(F)(F)F CC(C)C(CO)C(=O)NCCC1CSCCN1C(=O)CN1CCCCC1 C1(F)(CNC(C2(C#C)CCC2)=O)CCN(C(C2CC(CC)=NO2)=O)CC1 Cc1cc(C)c(C(N2CCCN(C(C3(c4cccnc4)CC3)=O)CC2)=O)c(Cl)n1 c1(OC)cc(C(=O)CCC(=O)NC2CC(NC(c3cc(C)c(C)s3)=O)C2)ccn1 C#CCCCC(C)C(=O)NCC1(CNC(c2cccc(O)c2Cl)=O)CCCCC1 C1(C(C)C)CN(C(=O)CCCCCF)CCN1C(c1cccc(C(C)(C)C)c1)=O c1(CNC(N2CCOC(c3nccs3)C2)=O)ccc(CO)cc1 Cc1cccc(C(=O)N(CC(C)NC(c2c(C)cnn2C)=O)C)c1[N+](=O)[O-] C(=O)(CCCCc1ccccc1)NCCN(C(=O)C(C)(CO)OC)CC N1(C(C(C)N(C(C2CC(O)(CC#C)C2)=O)C2CC2)=O)C2CSCC1C2 Cc1nc(C)c(CNC(=O)C(C)(CO)NC(=O)CCC2CC2(C)C)s1 C1(C(=O)NCC2(C#C)CCCC2)C2CCC(C2)C1NC(=O)C(C)N=[N+]=[N-] C(=O)(CC1OCCc2ccsc21)N(C)CC1CN(C(C(CC#C)O)=O)C1 c1(CC)ccc(C(=O)NC2CCC(CNC(=O)CSC)C2)s1 c1(NC(=O)Cc2ncc(-c3ccn(-c4ccccc4)n3)cn2)ncc(Br)cc1O N1(C(=O)C=CC2CCCO2)CC2CCCN(C(c3coc(Br)n3)=O)C2C1 Cc1cc(S(=O)(=O)NC(c2cc3ccc(F)cc3s2)=O)c(C)o1 Cc1ccnc(C)c1C(N1CC(CNC(=O)CC2CCC(F)(F)CC2)C(O)C1)=O Cc1ccc(CN2CC3(CC3C(=O)Nc3ncccc3F)C2)c(C)c1 N1(C(CCc2cc(C)[nH]n2)=O)CCN(C(c2ncc(N)cc2C)=O)C(C)C1C N1(C(CCN2CCN(CC)CC2)=O)CCCC(NC(C2(N(C)C)CCC2)=O)CC1 c1(C(=O)NC2CN(C(c3nc(OC)oc3)=O)C3C2C3)ccc(S(C)(=O)=O)s1 CC1CCC(C)N(C(C2CCCN(C(c3cnn4c3OCC4)=O)CC2)=O)C1 N1(C(C#CC2(C)COC2)=O)CCN(C(C2CCCCC2)=O)CC2CCCCC12 Cc1nc2ncnn2c(NCc2cnn(C)c2C)c1C C1(C(=O)Nc2cc(CC)[nH]n2)(CC)CCCN(C(C2CCC3CC2CO3)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NC1CC1NC(=O)CSC1CC1 C1(CNC(CSCCCC)=O)CCCCC1NC(c1ccc(OC(C)C)cn1)=O C#Cc1cc(F)c(C(N2CC(NC(=O)C=CC3CCCN3C)C(O)C2)=O)cc1F C(=O)(C(C)(C)CC(C)C)N1CC(SC)C(NC(=O)Cc2cscn2)C1 c1(C(N(C2CCN(C(C3OCCC3CC)=O)C2)CC)=O)ccc(F)cc1C c1(CN(C)CCNC(=O)CC2(N3CCOC3=O)CC2)nn(C)c(C(F)(F)F)c1Cl Cc1cccc(Cl)c1OCC(N1CCC(NC(=O)CC2(C)CCC2)C(CO)C1)=O N1(C(c2c(C)cco2)=O)CCC(CNC(C2CC(C)(C)C(C)(C)C2)=O)C(F)(F)C1 c1(COC(C)C)ccc(C(=O)NC(C)(C)C(C)NC(c2ccnc(S)c2)=O)cc1 C(C(C(=O)NCC1(CCCO)CC1)NC(=O)CCCc1ncco1)N(C)C C12(C3C(=O)NCC3)CC(CN1Cc1ccc(-c3ccccc3)s1)C2 C(=O)(C(F)CCC(C)(C)C)NC(c1cnn(C)c1)C(=O)NC1CC(C)CC1(C)C N1(C(Cn2c(C(C)C)ncc2)=O)CCC(N=c2nc(C(C)C)[nH]s2)C(C)C1 C(=O)(C1=CCCC1C)N1CCCC(CCNC(CCc2ccc(C)o2)=O)C1 C1(NC(C2(CC)CCC2)=O)CCC(C)(C)CC1CNC(c1cnn2c1OCC2)=O N1(C(C2(OC)CCC2)=O)CC2(C)CN(C(c3ccc(F)c(F)c3N)=O)CC2(C)C1 C1(NC(C(CC)C)=O)CCCCC12CCN(C(c1cccc3nn[nH]c13)=O)CC2 C(CC(=O)NCc1cnc(F)cc1C)(CC(C)C)NC(Cc1ccn(CC)n1)=O c1(NC(=O)NC2(NC3=NCCC3)CC(CO)C2)ncc(C(F)(F)F)cc1Cl c1(C(N2CC3CCN(C(C(C)SCC)=O)C3C2)=O)c(C)nn2c(C)cccc12 C1(NC(CNS(CC)(=O)=O)=O)CCCCN(C(=O)COCC2CCCC2)CC1 C(=O)(C(C)(C)c1csc(C)c1)NC1C(CNC(C2(SC)CCC2)=O)C1 C(CN=c1ccc2cccc(Cl)c2[nH]1)OC1C(=O)c2ccc(Br)cc2O1 CCC(C)(C)C(=O)N(C)CCC1CCCCN1C(c1csc(C(N)=O)n1)=O C(=O)(C(C)C(O)C(C)C)N1CC(N(CCCC)C(=O)C=CC(=O)NC(C)(C)C)C1 C1(NC(C2(F)CN(C(CN(C(C)C)C)=O)C2)=O)CC(C)OC1=O c1(C(=O)NCCCOCCN(C(CC(C(C)C)C)=O)C)cnn2c1CC(C)CC2 CC1(C(N2CCC(n3ccnn3)C2)=O)CCN(C(=O)Cn2cccnc2=O)C1 c1(CN(C(C(C2CN(C(C3(COC(C)C)CC3)=O)C2)O)=O)C)nccn1C c1(C(=O)NC2C(NC(C3N(CC)CCCC3)=O)C2)ccc2cc(F)c(F)cc2n1 c1(C(=O)NC(C(C(C)C)NC(=O)CCC(C)(C)F)C)nc2cc(O)ccc2[nH]1 CN1CCC2(CCN2C(=O)CN(C2CCC2)C(C2CC(=O)CC(=O)N2)=O)C1 c1(-c2cccc(C)c2F)cnc2c(C(=O)NCC3=CCCOC3)c[nH]c2c1 c1(CC)ccccc1C(=O)N(C)CCNC(=O)C(c1cnn(C)c1)OC CCC(CC)C(C(=O)N1CCCCC1CCCNC(c1ccc(Br)o1)=O)OC c1(OC(C)C(=O)OCc2conc2F)ccc2c(c1)CCC2 C(C(C)CC(=O)N1CC(C)(C)C1)NC(C(OC)OC)=O c1(OC)ccc(NC(=O)C(C2CCCO2)NC(=O)C(C#N)C(C)C)nc1C Cc1nc(C(N2CC3(C2)CN(C(=O)CC2CC4CCC2C4)C3)=O)cc(O)n1 C1(CC)C(NC(=O)CS(=O)(=O)NC)CCN1C(C1CC=CCC1)=O N1(CC)CCC(C(=O)NCC(O)C(=O)N2CCCC2COC(C)=O)C1 C12(CNC(c3ccc(CC)s3)=O)CC(CN1C(=O)CNC(=O)C(F)(F)C1CC1)C2 Cc1cccc(C(=O)NC(C(=O)NCCC2CCOCC2)C2CCC2)c1C#N n1(C2CCN(C(C(c3ccccc3Cl)N(C)C)=O)CC2)cnc2ccccc12 Cc1cc(C(N2CC3C(C2)N3C(c2cc(Br)ncc2Br)=O)=O)ccc1F C(C(C)(C)C(=O)NC1CC1)OCC.C12CCC1CNC2=O c1(C(=O)NCC(C)(C2CC2)NC(C2CC3(CCO3)C2)=O)cc(F)ccc1Cl N1(CC)CCN(CC(=O)NCC2(F)CCN(C(C3CNC(=O)C3)=O)C2)C(=O)C1=O c1(C(C)C)nnc2cc(NCC(CC(C)C)NC(=O)C(C)CC3CCC3)ncn12 CC1CN(C(=O)CC2CCC(C#N)C2)CCN(C(c2cc(F)ccc2CO)=O)C1 CN1CCN(C(C2CCS(=O)CC2)=O)C(CNC(c2cnc(S)nc2)=O)C1 C#Cc1ccccc1C(N1CC2(C1)CN(C(c1cccc(C)c1F)=O)C2)=O Cc1nc(C=CC(=O)NC2(CNC(C3CCC(C)CC3C)=O)CCC2)[nH]c1C C(CCC1CC1)(C(=O)N1CCC2CC12)NC(C=CC=CC)=O c1(N2CCC(N(C)C(C3(Cl)CC3)=O)C2)ccc(C#N)cn1 c1(C(C)SCc2ncc(-c3ccccc3)o2)cccc(Br)c1 C1(C(=O)NCCC(C)O)OCCC1NC(=O)C(C)C1CCCO1 C1(C(=O)NCC2C(N(C)C)COC2)CCN(C(C2CCC3(CCC3)O2)=O)CC1O c1(C(=O)NCC2(F)CC(NC(c3c(C(C)C)cco3)=O)C2)cnc(S)n1C CC(C)CCCC(=O)N1CCC(O)C1C(=O)NC(CN(C)C)CCO Cc1cn2ccnc(C(=O)NC3CC(NC(c4ccnn4CCF)=O)C3)c2n1 c1(NC(CNC2CC(CC)OCC2)=O)cc(Br)ccc1[N+](=O)[O-] CCC(CC(=O)NCCNC(C1CC=CCC1C(F)(F)F)=O)SC CC1=C(C(=O)NCc2cccc(NC(c3coc(Cl)n3)=O)c2)CCO1 N1(C(C2CCCN(CCC)C2)=O)CCC(C)(CNC(c2sccc2F)=O)CC1 c1(NC(C(=O)Nc2c(C)n(C(C)C)nc2)=O)ccc(I)c(Cl)c1 Cc1cc(=NC2CC(F)(CNC(C34CCCC(CCC3)C4O)=O)C2)c(C#N)c[nH]1 CC(CCC(C)(C)C)C(=O)NC1CCC1NC(c1ccc(Cl)c([N+](=O)[O-])c1)=O Cc1cccc(C(=O)NCC2(O)CCN(C(C3(O)CC3)=O)C2)c1O C=CC1(C(=O)NC(CC#CC)C(=O)OC)CCN(C(c2ccc(Cl)o2)=O)C1 CC1(C)CC(C)(CNC(C2CC2[N+](=O)[O-])=O)CN1C(=O)Cc1c(F)cccc1Cl C12(NC(=O)CSC3CCS(=O)(=O)C3)CCCN(C(c3cnsn3)=O)CC1C2 N1(C(c2c(C(C)C)cnn2C)=O)CCCN(Cc2ccccn2)CC1 C1(CNC(C(COC)OC)=O)N(C(C2C=CC=CC=C2)=O)CCC1(C)C Cc1ccc(Br)c(C(N2CCCCC2C2CCCN(C(=O)CCF)C2)=O)c1 c1(C(=O)NCC2C(NC(c3cnn(CC)c3Cl)=O)CCCC2)ccnc(O)c1F C1(CC)(CNC(=O)C=CC(C)(C)NC(C2CC(=O)C2(C)C)=O)CCC(=O)N1 N1CCC2CC(c3nn[nH]n3)C2C1.c1cc2sc(C3CCCCC3)cc2s1 c1(CC(=O)N(C(C)CCNC(C2CC2c2ccco2)=O)CC)ccc(OC)cn1 c1(C(N(C(CNC(C(CC)=CCCC)=O)C)CC)=O)nnn(C)c1C C(=O)(CCCC#N)N(C1CCCN(C(=O)Cc2cccc(C)c2)C1)CC N1(C(C(CC)=CC)=O)CCC2(CC1)CN(C(C1CCCN(C(=O)OCC)C1)=O)C2 CCCC(C(=O)NC1CC(C)(NC(C2CCC(C)(C)C2)=O)C1)OC Cc1cc(C)c(C(=O)NC2CC(C)N(C(c3ccncc3F)=O)C2)[nH]1 c1(C(C)C)ccccc1C(=O)NCC1(C(=O)NCC(C)(O)C2CCC2)CCC1 c1(C(=O)Nc2ccc(C#N)c(F)c2)ncc2ccc(Br)cc2n1 CCC(CNC(c1cn[nH]c1)=O)(CC)NC(c1cnn(CC(F)(F)F)c1)=O C1(C(=O)OC(C)(C)C)CC2C=CC1N(OC(=O)Nc1c(O)ccc(OC)c1)C2 c1(NC(C2CCCN(Cc3nc(C(C)C)on3)C2)=O)c(C2CC2)nc2sccn12 c1(CC)cc(C(N2CCOCC2CNC(c2cncc(Br)c2)=O)=O)nn1C c1(NCC(=C)CC)ncc(C)cc1S(=O)(=O)N1CCC(P(C)(C)=O)C1 C1(CNC(CC(C)OC)=O)CN(C(=O)C=Cc2cnccn2)CC(C)(C)O1 c1(OC(C)C)ccc(C(=O)NC2(C)CCN(C(C3CN(C)CCO3)=O)C2)cn1 C1(C(N(CCCO)CCC)=O)N(C(c2cc(C)cc(C)c2)=O)CCC1(C)C c1(NC(=O)C=Cc2ccc(-c3ccc(F)cc3)o2)cnnc(O)c1Br C(=O)(C1=NNC(C(F)(F)F)C1)NCC1(OC)CN(C(CCC(=C)C)=O)C1 CCC(C)C(C(=O)NCC1CC2(CCO1)CC2)NC(=O)C(C(C)OC)N(C)C CC1=C(C(=O)N(C2CCN(S(=O)(=O)CC3(C#N)CC3)CC2)C)CCCO1 CCC(CC(C)C)C(=O)NC12CC(C(N3C(CO)CCC3CO)=O)(C1)C2 c1(CC)cccc(CC)c1C(=O)NC1CCCCC1CNC(c1cnsc1C)=O N1(C(c2c(C)nn(C(C)C)c2)=O)CC2CC1CN2C(=O)COCC(F)(F)F c12ccc(cc1)C(=O)N(C)C2.c1(Nc2ccc(C)[nH]2)ccc(COC)s1 C(CC(=O)N1CC2CC(CO)C(C2)C1)(C(F)(F)F)NC(C1C2CCCC12)=O c1(C(=O)NC(C2CCCN2C(=O)C(C)=CC(C)(C)C)C)ccc(CCC#N)cc1 c1(C(C)C)ccc(C(=O)NCCC2CCCN(c3ncc(Br)cn3)CC2)c(O)n1 C1(C(N2CC(OCCNC(CC(=O)OC)=O)C2)=O)CC12CCOC2 N1(C(c2c(O)ncc(CC)c2)=O)CCC2(CCCN(C(=O)Cc3c[nH]nc3O)C2)C1 c1(C(=O)NCC2CCN(C(C(C(C)O)(F)F)=O)CC2)c(F)ccc2c1OCO2 c1(OC)c(C(N2CCN(C(c3ccsn3)=O)C(C)C2C)=O)cnc2c1cnn2C C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NC(CO)C(F)(F)F)(COC)C=CC1 C1(NC(C2C(C)OCC2)=O)CN(C(c2ccc(-n3cncn3)cn2)=O)CC1OC Cn1nc2cccc(C(=O)NC3(CCCNC(C4CCOC4)=O)CC3)c2n1 C1(C)(NC(=O)C(C)OC2CCCC2)CCCC1(F)F.Cc1cc2oc1C(=O)NC2 C1(C(=O)NCCC2CCC(NC(c3onc(C)n3)=O)C2)CCN(C)S1(=O)=O C12(CNC(c3cn(C)c(Br)c3)=O)CCC(C1)N(C(=O)CC1CCOCC1)C2 C1(CN(C(=O)CCN2CCCC2)C)CCN(C(C2CC2(c2ccccc2)C)=O)C1 N1(C(C(C)=CC2CC2)=O)CCCC1C(C)NC(=O)C=CC1CCC1 N1(C(c2c(N)nc(Cl)cc2)=O)CCN(C(=O)C(O)CC2CCOCC2)CC12CC2 N1(C(C(COC)(F)F)=O)CCC(C)(NC(C23CC(F)(C2)C3)=O)CC1 N1(C(c2c(C)nns2)=O)CCC2CN(C(=O)CC3CC4CCC3CC4)CC12 c1(C(N2CCC(c3ccccc3)(CO)C2)=O)scc(C(=O)O)c1Br c1(C(N(CC(CC)NC(c2nncn2C2CC2)=O)C)=O)nc(C(C)(C)C)cs1 C(=O)(C(C)(C)C(C)(F)F)N1CC(NC(C(C2CCCC2OC)OC)=O)C(C)C1 C(=O)(C1=NOC(CNC(=O)Cc2cscn2)C1)NCC(C#C)C(C)C N1(C(COC(CC)C)=O)CC2CC(C)N(C(c3cnn(C(F)F)c3)=O)C2C1 c1(CC)cc(C(=O)NCC#CCNC(=O)CCc2cncc(C)c2)c(C)nn1 c1(C(=O)OCC)sc(CCC(=O)NC2C=CCN(C(=O)OC(C)(C)C)C2)nc1C N1(C(c2ccc(N(C)C)c(F)c2)=O)CC(NC(c2coc(Cl)c2)=O)CC12CCC2 C1(C(N2CCC(N(CC#C)C(c3ccccc3Cl)=O)C2)=O)CCCCC(=O)N1 C1(C)(CNC(CCC(C)SC)=O)CN(C(c2sc(C)nc2C)=O)CCO1 Cc1cc(C(=O)N(C)CC2CC(F)CN2C(=O)Cn2nccn2)nc(N(C)C)n1 N1(C(CN(C(C)=O)C)=O)CC(NC(C2(C#N)CCOC2)=O)CC2(CCC2)C1 c1(CC)ccccc1C1CC1C(=O)NCC(C1CC1)NC(c1cccnc1Cl)=O C(=O)(C1CCNc2ccccc21)NC1CC(CNC(c2csnn2)=O)C1 Cc1cc(C(=O)NCC(C)(C)NC(=O)CC2(c3ccccc3)CCCO2)cnn1 C(=O)(C(CC(C)C)OC)NCC=C.c1(C2C(=O)OCC(C)N2C)nc(Cl)sc1Cl CC(C)C(C)C(C)CC(=O)NCCOCCCNC(=O)Cc1ccc(F)c(F)c1 C(=O)(C(C)CN(C)C(C1CCC(=O)C1)=O)NCC(c1ccncc1)C N1(C(C2=C(C)CCCC2)=O)CCCC(C2CC2NC(=O)COc2cnn(C)c2)C1 C1(NC(c2ccn3cnnc3c2)=O)CCN(C(=O)Cc2cc[nH]n2)C12CCCC2 N1(C(C=C(C)c2ccco2)=O)CC2(CCCC2NC(C2CC3CCC2C3)=O)C1 C1(NC(CC)=O)C2CCC(OC(C)=O)C2CN1C(=O)COCc1nc[nH]n1 CC1CC1C1CC1NC(=O)CCN(C(=O)COCC1CC1)CC1CC1 C12CC(=NO1)C(=O)NC2.C1(O)(CC#C)CC(C(N2CC=CCC2)=O)C1 C(=O)(C(C)(C)C(C)(C)C)NC(C1CCCN1C(c1ccnc(C#N)c1)=O)C c1(NC(c2cn(C)nc2OC(C)(C)C)c2n(C(CC)C)nnn2)cncc(Br)c1C C=CCC(C)(CC)C(=O)NCC1CN(C(=O)CNC=O)C(C)(C)C1 c1(C(N2CC(CNC(C(C=C)(C)C)=O)N(C)CC2)=O)ccc(OC)c(OC)c1Cl C(=O)(CC(F)(F)C(F)(F)F)NCC(CC=C)NC(c1cccn1C)=O C=CC1CCCCN1C(=O)C(O)CCCNC(=O)C1CC1 N12CCC(CC)C1C2=O.C(CN=[N+]=[N-])OCC.C12(CCC1)CC(=O)NCCO2 c1(OCC)cc(NC2(CO)CCCN(C(c3cc(F)cnc3Cl)=O)C2)nc(C)n1 C1(C(C)O)CCCCN1C(C1CC(CCNC(c2cc(Cl)ns2)=O)C1)=O C12(NC(=O)CC3COCCO3)CCCC1N(C(c1cc(F)c(Cl)cc1F)=O)CC2 Cc1ccc(C2(NCC3CC3NC(=O)CC(O)C3CC3)CCC2)cc1 c1(SC)cccc(N2CC3(C2)SCCC3NC(c2ccsn2)=O)c1[N+](=O)[O-] Cc1cc(NCC(C)NC(=O)CCc2ccncc2)ccc1[N+](=O)[O-] C1(OC(=O)NC2CCCC2NCc2n(C)nc(C(F)(F)F)n2)CCC(F)(F)CC1 C#Cc1ccc(C(N2CC3CC(NC(c4cnccn4)=O)C2C3)=O)c(OC)c1 C1(CC(N2CC(CC(C)NC(COCCCCCC)=O)C2)=O)CCCC(C)(C)O1 C1(COC)CC(N=c2nc(N(C)CCn3cnnc3)c3cc(F)cc(F)c3[nH]2)C1 c1(C(=O)NCC2CN(C(=O)Cc3cncnc3)CCO2)cc2ncc(Br)cn2n1 C1(C(N2CC(COC)(NC(=O)CNC(C)=O)C2)=O)CCC2CNCCN12 Cc1cc(C(=O)N(C2CCN(C(c3cc4cccn4cn3)=O)C2)C)cc(F)c1F C(CCCCCC(=O)N1CC=CCC1C(=O)OC)NC(c1ccn(CC)c1C)=O C1(C(=O)NCC2(O)CCN(C(C(C)CN(C)C)=O)C2)CC1C1CCCCC1 CCCCC(CNc1ncccc1C(=O)OC)NC(=O)CCC(C)c1ccccc1 C(CCCC(=O)NCC1CC1NC(=O)Cc1ccc(C(C)C)cc1)OCCC=C N1(C(C2CC(O)C2)=O)CC2CN(C(=O)CCCc3cccnc3)CCC2(CO)C1 C1(CNC(=O)CCC2CCCC2)CCC(C(=O)NCCc2nncs2)CC1 CC1CC(CN)CN1C(=O)C(=O)Nc1ccnn1C1CCOC1 Cc1cc(OCC(=O)NCCCCNC(=O)C#CC2CCOC2)cc(C)c1Cl Cc1ccc(C=CC(N2CC(NC(=O)Cc3cccc(Cl)c3)CC(C)C2)=O)cc1 C(=O)(C(CCC(C)C)NC(c1sccc1Cl)=O)NC1(C#C)CCCOC1 C12(C(=O)OC)COC(C(=O)NCCCCN(C)C(C3CNC(=O)C3)=O)(C1)C2 C1(NC(=O)CCC(F)F)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC1O N(C1CCCc2c(O)cccc21)CC1C(C)CCCC1 CCCC(C(=O)N(CC)CC)n1cccc1.C1(C(C)C)C(=O)O1 N1(C(c2n(CC)cc(Cl)c2)=O)CCC(C)C(CNC(=O)Cc2cnn(C)c2)C1 C1(C(=O)NC2(C)CC(NC(C(C)(Cl)Cl)=O)C2)CC(C2CCC2)C1 c1(CNC(=O)CC2COCCN2Cc2cnn(C(F)(F)F)c2)ccc(F)cc1O C(N=c1[nH]c(N2CCC3CCCC3C2)nc2c1CSC2)c1nccc(CC)c1 c1(C(N2C(C)CCN(C(=O)CC3SCCO3)CC2)=O)ccnc2c1nnn2C c1(CC#N)cc(-c2cc(N)ccc2Cl)cc([N+](=O)[O-])c1 C1(CNC(CSCC)=O)CCN(C(=O)CCOCC2CCCO2)CC1C C(CNC(=O)COCCCF)(C(=O)N1CCC1CC(C)(C)C)N(C)C C1(C(=O)NCc2c(C)n[nH]c2C)CCN(C(C2CCN(C)C2)=O)C12CCC2 c1(OC)cc2c(cc1COC(c1cccc3c1CC(C)(C)O3)=O)OC(C)C2 C12(C(=O)NCC3CCC(=O)O3)CC(CO)(CN1C(C1CC(O)C1)=O)C2 C(C)(C(C(=O)NCCC1CC(=O)C1)C(C)C)NC(C1CCN(CC)CC1)=O CCC(C(=O)N(C)CC1C2CN(C(c3cnns3)=O)CC12)C(C)(F)F CC1C(C(=O)N2CCC(N3CCN(C(C4(C)CC4(C)C)=O)CC3)CC2)=NOC1C c1(C(N2CC(NC(C3CCN(CCN(C)C)C3)=O)C2)=O)ccnc(C(C)(C)C)n1 C1(C(=O)OC)CCCN(C(C2(F)CC(NC(=O)NC)C2)=O)C1 C1(CNC(c2cc(O)nc(Cl)c2)=O)CCCCCN1C(C1CCOCC1)=O c1(CC(N2CC(CNC(C3CC(O)C3)=O)C(O)C2)=O)ccc(Cl)cn1 C(C(C)(C)C(C)(C)O)NC(C1CCN(C(c2ccc(OCC)o2)=O)C1C(C)C)=O C1(CNC(=O)C=CC2CCOCC2)CN(C(c2snnc2C2CC2)=O)CC12CC2 N1(C(C2(N(C)C)CC2)=O)CCC(O)(C2CCN(C(=O)CC(C)(C)C(F)F)CC2)C1 c1(C(NNC(=O)Nc2ccc(COC(C)C)cn2)=O)nc2c(s1)CCCC2 CC(C(F)C(=O)N1CCC(=O)N(CC(F)(F)F)C1)C(F)(F)F C(C1CCCn2c(C)cnc21)Nc1nc(C)nc(NC2CSC2)c1 C(=O)(C(O)CNC(=O)C(F)=C(C)C)N1C(CC)CC1 C1(NC(C2CCN(CC)C2)=O)CN(C(C2(C(C)C)CNC(=O)C2)=O)CC12CC2 c1(CC)ccc(O)c(C(N2CC(CNC(c3nnsc3C)=O)C2)=O)c1 N1(C(c2c(OC)cccc2F)=O)CC(NC(C2CC2CF)=O)CC12CCCC2 C1(C(=O)NCCNC(CCCN(CCOCC)C)=O)CCCC12CCC2.OCC CC(O)C(C)CNC(c1ccoc1CNC(C1CCN1C(C)(C)C)=O)=O C1(CC)CCC(C)CN1C(C1CC(OC)CN1C(=O)C(C)SC)=O N1(C(c2cccc(C(C)(C)C)c2)=O)CC2CCC(C1)N2C(C1(C)CCOC1)=O c1(C(N(CCCNC(c2cccc(Cl)c2)=O)CC)=O)cnn2c1S(=O)(=O)NCC2 C(N=c1nc(C2CC2)[nH]s1)C1OCC(CNC(c2cc(-c3cccs3)[nH]n2)=O)C1 CCC(C)CC(=O)NCCN(C1CCCCCC1)C(=O)CCNC(=O)CC N1(C(CCc2ccc(C)s2)=O)CCC(C)C(NC(=O)CC2CCCNC2=O)C1 C1(C(=O)N(C)CC2(O)CCN(C(c3nnnn3C)=O)C2)(SC)CCC(F)(F)CC1 C(C)(C)(CCC(=O)NCc1ccc(C(=O)NC2CCOC2C(C)C)cc1)OC N1(c2c(Br)cnc(OC)n2)CCC(C)(C)C(CNC(=O)CSc2nncn2C)C1 C(=O)(C1=COCCO1)NC(C1CN(C(C2CCCC(C(=O)OCC)C2)=O)C1)C C(=O)(C1CCc2cc(F)ccc21)N1CC(C)(NC(C2CC(O)C(F)C2)=O)C1 CCC1=C(C(=O)NC2CC(CNC(C3CCC(C)NC3=O)=O)C2)SCCO1 C(C(N=[N+]=[N-])C(=O)NC(CCF)C(=O)NCc1ccc(C#N)cn1)OCC C1(N=[N+]=[N-])(C(=O)Nc2cc(C)sc2C)CCN(C(=O)C=Cc2cnn(C)c2)C1 C1(=CC(=O)NC(CNC(C2C(C(C)=O)C2(C)C)=O)CO)CCC(C)CC1 c1(C(=O)OC)ccc(NC(C)CC(C)(C)OC)c(F)c1 C=CCC(CC(C)C)C(=O)NCC1CCCC1NC(c1c[nH][nH]c1=N)=O CN1C(=O)CSC1=CC(=O)NC(c1ccccc1)CNC(=O)CCc1ccn(C)c1 Cc1ccc(CN2CC3(CC3)CC2C(=O)Nc2cc(Br)cnc2Br)cc1C N1(C(=O)COc2cccnc2Cl)CC2CN(C(C3(CF)CCC3)=O)CC2C1 c1(NC(C2CC(=C)CN2Cc2c(C)cccc2Cl)=O)cnc2ccc(Cl)nn12 C1(NC(c2c(C)onc2Cl)=O)CCN(C(c2cnc(=N)[nH]c2)=O)C(C2CC2)C1 N1(C(C(COC)O)=O)CCC(C2CCCN(C(c3cc(S(C)(=O)=O)co3)=O)C2)C1 C1(C(=O)NC2(CO)CCN(C(C34CCC(C)(OC3)C4)=O)C2)CCc2n[nH]cc2C1 c1(OC)ccc(NC(c2cnc(Cl)[nH]2)=O)c(C)c1.N12CC(CC1C)C2=O N1(c2nnc(C)s2)CCC2(COC(CNC(C3CCn4ccnc4C3)=O)C2)C1 C1(C(=O)NC(C)Cc2cn[nH]c2)CCN(C(C2CCCCC2)=O)CCO1 c1(C(=O)NC(CNC(C2C(C(=O)OC)C2)=O)C(C)(C)C)ccnc(F)c1OC c1(C(N2CCCC(CCNC(=O)Cc3ccon3)C2)=O)cc(=O)n2ccsc2n1 C1(NC(C(=O)NC(C)C)=O)CN(C(=O)CC2CCN(CC(F)F)CC2)C2CC12 N1(C(c2n3c(nn2)SC(=C)C3)=O)C2CCC1CN(C(c1nn(C)nc1C)=O)CC2 c1(OCC)ccc(NC(C2CSCN2C(c2ccc(O)cc2)=O)=O)cc1 Cc1c(C#N)c(N2CCC(n3cc(COC(C)(C)C)nn3)C2)nc2ccccc12 c1(C(N(CCNC(=O)CCc2ccc(Cl)s2)CC)=O)cncc(F)n1 c1(C(=O)NCCC(C)(C)NC(c2cncc(N(C)C)n2)=O)c(N)cc(Cl)cc1F c1(C(=O)NCCCCCCN(C(=O)C=CCn2cccn2)C)cc(O)nc(Cl)c1 c1(C(=O)NC2(COC)CN(C(C3(C)CC=CCC3)=O)C2)ccc(F)c(C(F)F)n1 c1(NCC(=O)NC(CC)CNC(C2CC2F)=O)ccc(C(N)=O)cn1 c1(OC)cc(C(=O)NCC2CC2NC(C2CC3(CCCO3)C2)=O)cc(F)c1F CN1N=C(C(=O)NCC2CN(C(C34CC(C#N)(C3)C4)=O)C2)CCC1=O c1(OC(C)C)cccc(C=CC(N2CC(F)(CNC(C3CCCOC3)=O)C2)=O)c1 Cn1cncc(C(=O)NCCCC(N2CCOC3CC23)=O)c1=O c1(CC)sc(C(=O)NCCOCCNC(c2coc(C)c2)=O)cc1C C1(NC(C2(NC(C3C(C(N)=O)COC3)=O)CC(F)C2)=O)CCC(C#N)CC1 C(=O)(C1CCCc2ccnn21)NC(C1(O)CCN(C(C(CC)=CCCC)=O)C1)C Cc1cc(NC(c2c(Br)n[nH]c2C)=O)ccc1NC(c1ccnn1CCF)=O N1(C(C2(C)CNC(=O)C2)=O)CCc2[nH]nc(CNC(C3CC=CC3)=O)c2C1 CC1(C)NC(=O)CCC1NC(=O)CCOCCNC(=O)COC1CCC1 N1(C(C(CC)C)=O)CCC(NC(=O)CCCc2ccccn2)C1CC C=CC(C)(C)C(=O)NC1CC(CCNC(c2conc2C(C)C)=O)C1 NC(=O)CCCC(=O)NCC(=O)NCc1cn(C2CC(O)C2)nn1 c1(C(=O)NC2(COC)CCCOC2)n[nH]c2c(C(=O)O)cccc12 C1(C(C)NC(COCC(C)C)=O)CCN(C(c2cnn(-c3cccnc3)c2)=O)C1 c1(CC)cc(C(=O)NCC(C)(CO)NC(=O)C(O)Cc2ccccn2)c(C)nn1 c1(CCC(C(=O)NC(C)(C)C)N(CCOC)C(C)C)ccc2ccccc2n1 c1(C(=O)NCC2CN(C(C3(SC)CC(O)C3)=O)C2)cccc(C#N)c1 CC1(C(=O)NCC2CC2CNC(=O)Cn2nnc(=N)[nH]2)CCCCC1(F)F c1(C(=O)NCCCC(C)NC(C2C(C)C2)=O)ccccc1C(C)(C)C#N Cc1ccc(F)cc1CCNC(=O)NCC1CCN(S(=O)(=O)c2cccs2)CC1 C12(CNC(c3c(C)ccc(C)c3)=O)CCCC1N(C(=O)Cc1ccoc1)CCC2 C(CC(CC)C(=O)NCCCOCCC(N1CCOC(C)CC1)=O)=CC CCC(C)C(=O)NC(Cn1cccn1)C(=O)N(C)CCn1cnnc1 O=C1CC(CC(N2CCCC(NC(=O)CCC3CC3)C2)=O)C(=O)N1 Cc1ccc2ncc(C(=O)N(C)CCN(C)C(C3COC(C)(C)O3)=O)cc2c1 c1(NCC2CCN(C(=O)OC)CC2)nccc(=NCC2=COCCO2)[nH]1 CC(C)CS(=O)(=O)N1CCC(CC(=O)NCCCC2(C)OCCO2)C1 C(=O)(C(C)CC(N)=O)NC(C(=O)NC1C(CN(C)C)C1)Cc1ccccc1Br C(=O)(CCCC(=O)C1CC1)N1CCCC(OCC(N2C(C)CC2CO)=O)C1 N1(C(C=C)=O)CCCC(C(N2CCC(NC(c3cccnc3)=O)CC2)=O)C1 CC(C)CCC(=O)C(=O)NCc1cc(C(=O)NC(c2cccnc2)C)no1 c1(C(=O)OCC(c2cn(C)nn2)=O)ccc(CCNC2(C)CCC2)cc1 c1(C(=O)NC(C)C(C)NC(C2(F)CCCCCC2)=O)ccc(S(N)(=O)=O)cc1 c1(C(N2CCN(C(C(CC=CC)CC)=O)C(CCC)C2)=O)cc2sccc2n1C c1(C(N2CCN(C(c3ccn(C)n3)=O)C3C2C3)=O)cc2cc[nH]c(=O)c2s1 N1(C(C)=O)CCCN(C(c2cnn(C)c2)=O)CC1 N1(C(CCC(=C)Br)=O)CCN(C(c2cc(C)c(N)cn2)=O)C(CO)C1 C1(OC)(CO)CCCN(C(=NCC(C)C)NCc2c(C)nn(C(C)C)c2C)C1 C(=O)(CC(CNC(C1COCOC1)=O)C1CCC1)NC1(CC(=O)OC)CCC1 C1(CNC(c2cnc(OC)s2)=O)C(C)CCCN1C(=O)C(O)CC1CCCC1 C1(C(=O)NCC2N(C(C3CCCC(=O)N3)=O)CC=C2)CC12CCCCC2 N1(C(C(C)Cn2ccnc2)=O)CC(N=[N+]=[N-])CC1C(=O)NC(C)Cc1nc[nH]n1 C1(CNC(CC(C2CC2)NC(C(C2CC2)SC)=O)=O)CCN(C2CC2)C1=O c1(CC(CNc2cc(OCC)nc(COC)n2)CO)ccc2nonc2c1 C(=O)(C(C)(F)C(F)(F)F)NC1CN(C(c2ccc(OC)c(Br)n2)=O)C1 C(=O)(C1=CCN(C(c2cccc(Cl)c2)=O)C1)NC(CC)COC C(=O)(CC(C)C(C)(C)C)NCC1C(NC(CCCCOCC)=O)C1 C1(N(C)C)COCC1C(=O)NC1C(C(=O)NC(c2cn(C)cn2)(C)C)C1(C)C C#Cc1ccc(C(=O)NCC2(O)CCCN(C(=O)CN(C3CC3)CC)C2)c(F)c1 N1(C(C(C)=CC)=O)CC(C)CN(C(c2cccc3c2CCO3)=O)CC1C C=CCC(CNC(c1nc(Cl)oc1C)=O)C(=O)N1CC2C(C1)C2(C)C c1(C2(CNC(N(C)CC3CC3)=O)CCC2)conc1C(C)(C)C N1(C(C2(OC)CC2)=O)CCCOC(CNC(C2(C)CCNC2=O)=O)C1 Cc1nc2[nH]c(C(N3CCC(NC(c4c[nH]cc4C)=O)CC3)=O)cc2s1 C1(C(=O)NCCN(C(=O)C=C(C)C(C)C)CC)CCCC1Nc1ccccc1 C1(NC(COc2cn(C)nc2)=O)CN(C(=O)C(C)(C)F)CCC1CO N1(C(CN(CC(=O)NC2CC2C(=O)NC(C)(C)C)C)=O)CCCC(F)C1O N1(CC)C2CCC1CN(C(C1CCC(C)N1C(c1cccc(O)c1)=O)=O)C2 c1(COC)nc(C(=O)NC2CC(CNC(c3c[nH]nc3C3CC3)=O)C2)n[nH]1 N1(C(c2c(CC)nns2)=O)CC2CC1(CNC(C1(C)CCOC1C)=O)C2 N1(C(c2occ(C)c2)=O)CCC(NC(C2NC(=O)C3CC23)=O)CC(C)(C)C1 Cc1cc(C(=O)NCC(C)(C)NC(=O)Cc2cscn2)cnn1 N1(C(C2C(NC(Cn3c(C)ccn3)=O)CCO2)=O)CCC(C2=NOCC2)C1 c1(CCNC(c2nccs2)=O)n[nH]cc1C(=O)NCC1(CO)CCC1 C1(CNC(c2cc(Cl)c[nH]2)=O)(CO)CCN(C(=O)CC2CCOC2=O)CC1 C(=O)(C(C)CC(F)F)NC(CNC(Cn1nc(C)c(Cl)c1)=O)C1CCC1 CC1(NC(C2CC23CCC3)=O)CCC(NC(c2ccnn2C(F)F)=O)CC1 C(=O)(C1CCCc2ncnn21)NC1COCCN(C(CCC(=O)OC)=O)C1 O=C(C1CCCc2scnc21)NC1CCC2CN(c3nc(CC4CC4)ns3)CC2C1 c1(NC(C(=O)NC(c2ccccc2)C)C)nc(C(F)(F)F)n[nH]1 c1(C(=O)NC2C(C)N(C(=O)CN(C)C)CC2)c(-n2cnnn2)sc2c1CCC2 C1(NC(c2cc(F)cc(F)c2)=O)CCCCN(C(=O)Cc2csc(Cl)c2)CC1 N1(C(c2c(C)c[nH]n2)=O)CCCC2(C1)CN(C(C1CCCO1)=O)CCO2 c1(CN=C(NC(C2(CO)CCCC2)C)NCC2CC2)ccc2c(c1)NC(=O)CO2 Cc1ccc(O)c(CNC2CCC(CC(=O)Nc3c(C)cccc3F)CC2)n1 N1(C(c2n(C)ncc2C2CC2)=O)CC2(CC(NC(C3(CO)CCCCO3)=O)C2)C1 N(C)(C(=NCCCF)NCC1N(CC)CCOC1)CC1CCN(C(C)=O)CC1 C1(CC(=O)NC2CC(O)(CNC(c3cnc(Cl)s3)=O)C2)CCC12CCC2 c1(C(=O)NC2(C3CN(C(CCOC(C)C)=O)C3)CC2)cc2c(O)cccc2[nH]1 Cc1coc(C(=O)N(C)CC2CCCCN2C(C2C(C)(C)C2(F)F)=O)c1C C(=O)(C(O)CC(C)(C)C)N(C)CC1CN(C(c2nnc(S)n2C)=O)CC12CC2 c1(OC)cncc(C(=O)N(C(C)CN(C(=O)CCCc2ccccc2Cl)C)C)c1 N1(C(CS(=O)(=O)NC)=O)CC2CCC1C(NC(=O)CCCCC1CC1)C2 N1(C(C2C=C(C)CS2)=O)CCC(C2CCN(C(=O)C(C)(C)n3ccnn3)CC2)C1 C(CCCCC(=O)Oc1ccc(-c2nnc(OC)s2)cc1)n1cc(COC)nn1 C1(O)(C(=O)Nc2cccs2)CN(CC(=O)NC2C(NC(C(C)=C3CC3)=O)C2)C1 C1(N(C(CN2CC(C)(OC)C2)=O)C)CCC(NC(C2(C(F)(F)F)CC2)=O)CC1 C1(NC(C2CCCCC2O)=O)CCCC2(C1)N=N2 CC1(NC(=O)CC2CCC(=O)O2)CCCN(C(C2CN3CCN2CC3)=O)C1 c1(SC)ccc(C(C)NC2CN(CCOc3ccccc3)C2(C)C)cc1 C1(CC(=O)NC(C(C)C)CCN(C(=O)CSCC(N)=O)C)SC2=NCCN2C1=O c1(C(=O)NCC23C(CN(C(C(=O)C=Cc4cccs4)=O)C2)C3)ccc([N+](=O)[O-])cc1 c1(C(=O)Nc2cccc(CS(C)(=O)=O)c2)cc(C#N)ccc1Cl CCC(C#N)C(=O)N1CCC(COCCN(C)C(C2(NC(C)=O)CCC2)=O)CC1 c1(C(N2C(C)CCC(NC(C3(CN(C)C)CC3)=O)C2)=O)cnn2ncccc12 CCC(CC)C(F)C(=O)NC12CCC(C(=O)NC3CSC(C)C3)(CC1)C2 C1(CC(=O)NC2C(NC(=O)Cc3csnn3)CCCC2)CCc2ccccc2C1 CC(C)C(C(=O)NCCCCCN(C)C)C(C)NC(c1cc(C(N)=O)[nH]n1)=O c1(CC)cccc2c(C(N3CC(F)(CNC(c4cc(O)nn4C)=O)C3)=O)c[nH]c12 C1(NC(C2(S(N)(=O)=O)CC=CC2)=O)CCCC2CN(C(=O)C=CI)CC12 C(C1NCCc2sccc21)NC(=O)Cc1ccc(C(=O)O)cn1 c12ccnc(c1)OCCN(C(N)=O)CCNC2=O.CN1CCC(C(=O)OCCO)C1 CCN=C(NCCOC1CCOC1)NCC(C1CCCCC1)OC N1(C(C(CC)=CC)=O)CCC(NC(c2cc(F)c(F)cc2Cl)=O)CC(O)C1 N1(c2cc(OC)ncn2)CCC2(CCN(C(C3CN(C)C3)=O)CC2)CC1 N1(C(C2=CCC(C)CC2)=O)CCCC2(CCN(C(c3cscc3C#N)=O)CC2)C1 Cc1cc(C(=O)NCC2CN(C(c3cnsn3)=O)C(C)(C)C2)ncc1CO CC(CC(N)=O)C(=O)N1CCOCC1CN(C(=O)CCC1CCCCC1)C c1(C(N2CCN(C(C3(CO)COC3)=O)CC23CC3)=O)nccc2cccnc12 c1(C(C)NC(C(C)C2CCCC2)=O)nocc1C(=O)NCCc1cn(C)nn1 C1(C)(CC)CN(C(=O)C(CNC(C2CC2C#N)=O)OC)C1 C1(NC(C2C(C)CN(C(C3CC4CCC4C3)=O)CC2)=O)CC(C)(C)OC1(C)C C(C)(CO)(C(=O)N(CC(C)(C)C(=O)NCC(O)Cn1cccn1)C)OC C1(C(=O)NCCCCC2CN(C(=O)Cn3cncn3)C2)CS(=O)(=O)CC12CC2 c1(SC)cc(-c2ccc(C(=O)NCc3ccns3)nc2)ccc1F C1(O)(C(C)NC(C(C2CC2)OC)=O)CN(C(=O)CC2CC(C)(C)C2)C1 CCCC(C)(C)C(=O)NCc1ccc(CCCNC(=O)COC)cc1 c1(C(N2C(C)(C)CC(NC(C3CCC3C(F)(F)F)=O)C2)=O)cc2ccccn2c1 Cc1cc(Br)c(C(=O)NCCC2(CNC(c3cnc(S)[nH]3)=O)CC2)s1 C1(C(=O)NCC2CCN(C(=O)Cc3ccsc3)C2)CCC2CC1CO2 N1(C(CNS(CC)(=O)=O)=O)CCC(COC)(NC(=O)CCc2cccn2C)C1 CC1CC(CNC(=O)Cn2ncnn2)CN1C(c1ccc(CC(C)(C)C)cc1)=O N1(C(C2(NC(C)=O)CCC2)=O)CC(NC(=O)CCC(F)(F)F)CC(C)(C)C1 CC(c1ccccc1)=CCO.N12CCCC1SCCC2=O CC(C)(CCCCNC(=O)C(O)C1CCCC1)C(=O)NNC(=O)c1n[nH]cc1Cl C(=O)(C(C)CS(C)(=O)=O)NC1C(NC(Cc2c(C)ncs2)=O)CC1 C1(N(C(CCNC(C)=O)=O)C)CN(C(=O)C=Cc2ccnn2C(C)(C)C)CC1O C(=O)(C(C)C(C)NC(=O)CC1CC2C=CC1C2)OC.C1(C2CCC2)CC(=O)N1 Cn1ncc(C(=O)NC2CC=CCC2C(N2CCC2C2CCOCC2)=O)c1N N1(C(CCC(CC)OC)=O)CCC2C(CCCN2C(c2cc[nH]c(=NC)c2)=O)C1 c1(C(C)NCC2C(C(N3CCn4nccc4C3)=O)C2)ccc(S(C)(=O)=O)cc1 C1(C(=O)NCC2C3CN(C(c4cc(CO)c(C)o4)=O)CC23)(COC)CCOCC1 N1(C(C(c2ccccc2)OC(C)=O)=O)CCCC(N(C(=O)CS(C)(=O)=O)C)CC1 N(C1COCc2cc(Br)ccc21)C(=O)NCCCc1c(F)cccc1F C(C(C)(C(=O)NCC1CC1(C)C)NC(c1c[nH]c(C(N)=O)c1)=O)SC C12CCOC1C1CC1C(CC)C(C)C(C)NC(=O)COCCNC2=O c1(C(=O)N(C2CC3(CNC3)C2)CCCn2ccnc2)cc2n(n1)CCCC2 N1(C(C2C(C)(C)C2)=O)CC(CNC(c2cc(Cl)c(F)cc2O)=O)C2(CCC2)C1 c1(C(=O)NC(COCC)C(=O)NC(CO)CCSC)cc(C)nc(C)c1 CC1CN2CCN1C(C(N1CC(C(C)NC(c3ccc(C(C)(C)C)s3)=O)C1)=O)C2 CN1CCC(C(=O)NC2CCC(F)(CNC(c3nnn(C)c3N)=O)C2)CC1 c1(C(=O)NCCN(C(C2CCC(CC)O2)=O)CC)cnn(C2CCOCC2)c1C c1(C(=O)NCCN(C(CN(C2CC2)CC)=O)C2CC2)ccc(F)cc1C#N N1(C(C2CCCCO2)=O)CC2CCN(C(c3ccc(Br)cc3Cl)=O)C2C1 CC1(NC(=O)CC2(CO)CCOCC2)CCCN(C(C2CCC2)=O)C1 c1(C(N2C(CC(=O)NC3C(C#N)CCC3)CCC2)=O)ccc(Cl)cc1 C1(C(=O)NC2CCC(CO)C2)CC2(CCN1C(=O)CCF)CC2 c1(C(=O)NCc2cccc(C(=O)NCCC3CCCC3O)n2)cc(F)cnc1O C#Cc1cccc(C(=O)NCC2C(C)CCCN2C(=O)CC2CCC2)c1 C(C(C(C)C)NC(=O)Cc1ccsc1Cl)(c1ccccc1)NC(C1CC(=C)C1)=O CN(C)NC(=O)CCC(=O)N1CC2CC(NC(=O)CC(C)(C)CN(C)C)C(C2)C1 C(=O)(N=c1c(C)c[nH]cc1Br)C1C(NC(c2cc(OC)c(O)cc2)=O)C1 N1(C(CSCCOC)=O)CCC2C(C(=O)NCC(C)C(F)(F)F)C2C1 C(CC(C(C)C)NC(c1c[nH]nc1F)=O)N(C(C(CC)OCC)=O)C N1(C(C(C)NC(=O)C(C)(C)C2(O)CCC2)=O)CC(F)CC1C CCC(CC)(CCNC(c1ccn(C2CC2)n1)=O)NC(c1nc(C)sc1C)=O c1(C(=O)NC2CC3CC(NC(C(C4CC4)SC)=O)CC32)cc(C)cc2nc[nH]c12 C=CCCCCCC(=O)N(CC(C)O)CCNC(c1cnn(C)c1)=O CCC(F)(F)C(=O)NCC1(CC(N2CCC(OCCF)C2)=O)CCC1 C(=O)(C#CC1(C)CC1)N(CCCOCCNC(C(C(C)C)OC(C)=O)=O)C c1(C(=O)NC(CC)CC(=O)N2CCOCC2C2(C)CC2)cc2occc2[nH]1 C(=O)(C(C)(C)c1cc[nH]n1)NC1C(C(=O)NC2(C(=O)OC)CC2)C1 c1(C(=O)NC2CCCC(NC(C3N(C)CC(O)CC3)=O)C2)ccc2nncn2c1 C1(CN=C(NC(C=C)C)NC2CN(CCOCC)CC2C)CCCS(=O)(=O)C1 N1(C(CN(C(C)=O)C)=O)CCCC2CN(C(c3cnc(S)n3C)=O)CC12 C#CCC(C)(CC)C(=O)NCC(C)(C)CC1CN(C(c2ccncc2Cl)=O)C1 C#CCCCC(C)C(=O)NC(C1CCCC1)CNC(=O)Cc1cccs1 C1(CC)CN(C(=O)C=Cc2ccc[nH]2)CCN1C(c1cc(OC)cs1)=O c1(C(N(C2CC=CC2)CC)=O)ccc(C(F)(F)F)cc1.C12CCCC(C1)NC2=O c1(CCOC)cn(CCCN(C(C2CC2F)=O)Cc2occc2C(=O)O)nn1 C1(NC(CC)=O)CCC2(CC1)CCN(C(=O)CC1CCC(O)C1)CC2 N1(C(c2nccc(C)c2)=O)CC2CCC1CN2C(c1cc(Cl)c(F)cc1F)=O C1(NC(C(CC)COC)=O)CC(C)CN(C(=O)CCOc2cccc(C)c2C)C1 N1(C(c2nc(CCC)oc2)=O)CCC(C2CCCN(C(=O)C(O)C3CC3)C2)CC1 c1(C(=O)NCC(CC=C)NC(c2ccnc(CC)c2)=O)c[nH]cc(C)c1=O c1(CC(=O)N(CC(C)NC(=O)C(C2CC2)N(C)C)CC)csc2nc(C)cn12 N1(C(C2(CN(C(C(C)(C)OCC)=O)C)CC2)=O)CC2(CCN(C(C)=O)C2)C1 c1(C(N2C(CN(C(=O)Cc3cn(CC)nn3)CC)CCC2)=O)cc([N+](=O)[O-])n[nH]1 C1(NC(=O)NCc2c(C)ocn2)CCCN(CCNC(=O)C(F)(F)F)C1 c1(C(=O)OC)no[nH]c1=NC(=O)Cc1ccc(C(=O)NCCC(C)(C)O)cc1 C=CC1(CC(N2CC(N3CCCC3)C2)=O)CN(C(C2(C(C)=O)CC2)=O)C1 N1(C(c2c(OC)scc2)=O)CC2CCC2(CC(=O)N(C)CC2(C#N)CCC2)C1 c1(N2CC(C)(OC)OCC2)nc(=NCC2CC3CC3C2)[nH]c2c1CCC2 C(CNC(c1ccc(CCNC(=O)NC)cc1)=O)(CC(C)C)N(C(CC=C)=O)C C=CCC(CC(C)C)C(=O)NCCCCN(C(=O)C(c1ccc(F)c(F)c1)C)C C1(C(N(CC(C2CCC2)OC)C)=O)CC(O)CN1C(=O)CC1CCC1 C1(CC(C)NC(C(C)=C2CCC2)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(C)C CC1CCCC=C1C(=O)NC1(C2CN(C(C3(C)CCC3)=O)C2)CC1 C1(NC(C(C)(C)F)=O)CCN(C(c2cc(C(F)(F)F)ncn2)=O)C12CCC2 C1(NC(C2CCC(=O)NC2)=O)CC2CC(C1)N(C(=O)Cc1cc[nH]c1)C2 CN=c1[nH]c(SC)ncc1CN1CC(F)(C(=O)Nc2nc(Cl)ccc2Br)C1 CC(CN=c1[nH]c(C#N)c(Cl)s1)(C1CC1)NC(c1ccc2c(c1)CCOC2)=O C12(CC)CCC(C(=O)NC3CCC(CNC(C4(c5cccs5)CC4)=O)C3)(CO1)C2 C=CCC(CC)C(=O)N(C1CCN(C(=O)CCOCC(F)(F)C(F)F)C1)C CC1CCCC(NC(=O)OC(C)(C)C)CC1.N12CCCC(C1)C2 C#Cc1ccc(C(=O)NCC(C)(C)CN(C)C(C2CC23CC3)=O)c(OC)c1 C1(CCOC)CC1NC(=O)C=C(C)CNC(=O)CC1(CO)CC1 N1(C(C2C(C=C)C2)=O)CCN(C(=O)C=C2CCCCC2)C(CC(F)(F)F)C1 C1(C(=O)NC(C2CC2C(=O)NCCc2ncc[nH]2)C)CCOC1 C1(NC(N)=O)CCC(n2cccc2)CC1.C12(CCCC1)C(=O)NC2 C1(CNC(c2ncc[nH]2)=O)CCN(C(=O)COc2ccc(CO)cc2)CC1(F)F N1(C(C2CCCN(C(CSC(C)C)=O)C2)=O)CCC(C(N)=S)CC1 C1(CCC(=O)NC2CCC(NC(c3cc[nH]c3)=O)C2)CCOC1=O C1(NC(c2cccc3cncn23)=O)CCC2CC1CN2C(c1ccncc1F)=O C12(CNC(c3c(C)noc3)=O)CC(C1)C(NC(C1CCC(C)O1)=O)CO2 N1(C(C2(CC(C)C)CC2)=O)CCCCCC(NC(C2(F)CCS(=O)(=O)C2)=O)C1 CCC(C)(C(=O)N1CC(NC(=O)OC(C)(C)C)C(c2ccccc2)C1)OC CCCCCCCC(=O)NC(c1csc(C)c1C)c1nnnn1C(C)(C)CC c1(C(N2CC(NC(CC=CC=C)=O)C(F)CC2)=O)cc(Br)cc2c1OCC2 C1(CN(C(CSCC(=O)OC)=O)C)CCCCN1C(=O)C=CC1CCOC1 O=C1CC2(C1)CC(C(=O)NC1(C(=O)NCC3CC3C3CC3)CSC1)C2 N1(C(c2c(CC)scc2)=O)CCC(CNC(=O)C=CSCc2ccco2)C(C)C1 N1(C(CSc2n(C)cnn2)=O)CCC(CCNC(c2cc(C(N)=O)co2)=O)CC1 C12(CNC(c3ncc(CC)s3)=O)CCCCC1N(C(=O)CC(F)(F)C(F)F)CC2 C1(NC(c2c(CC)con2)=O)CC12CCN(C(=O)CC1CC1(Cl)Cl)C2 C1(N(C)C(C2CSCCS2)=O)CC2CC1N(C(c1cc(C(F)F)ccn1)=O)C2 c1(C(N(CC(C)(C)NC(C(C2CCC(=O)N2)C)=O)C)=O)cc2ccccc2s1 c1(C(N(C)CCNC(C23COC(CF)(C2)C3)=O)=O)c(Cl)cccc1Cl C1(NC(c2ccnnc2)=O)CN(C(C2(F)CC23CCCCC3)=O)CC2(CCC2)C1 Cc1c(C)c(C)c(CNC(c2nc3ccccc3s2)C(F)(F)F)c(C)c1C c1(C(N2C(CNC(CC(C)C3CCCCC3)=O)CC(F)C2)=O)ccnc(O)c1F Cn1nccc(C(N2CC=CC(NC(C3CCCCS3(=O)=O)=O)C2)=O)c1=O C1(CC(=O)NCCS(CC)=O)CCCN(C(c2ccc(F)nc2)=O)CC1 C(=O)(C(=O)CCC(C)C)N(CCOCCN(C(c1cncc(CC)c1)=O)C)C N1(C(c2ccc(NC)cc2)=O)CCCCCC(NC(c2c(C)occc2=O)=O)C1 C1(NC(c2c(C)nc[nH]2)=O)C2CC1N(C(c1ccc(OCC3CC3)cc1)=O)C2C c1(C(=O)Nc2cccc(NC(CCCCC)=O)c2)c(C)ccc(C)c1C(=O)OC c1(C(N(CCSC)CC)=O)cc(F)c(C)cc1N.n1(C)cc(CC(CO)C2CC2)nn1 N1(C(CSCCC)=O)CCC(NC(=O)C=Cc2ccc(Cl)cc2)C12CC2 C1(NC(c2scc(C)c2)=O)C2CCCN(C(C3CC4CC(=O)C3O4)=O)C2C1(C)C C1(CC(=O)NCCN(CCC)C(c2cc(C(F)F)[nH]n2)=O)CC(O)C1(C)C c1(C(=O)NCC2(F)CC(CNC(C=C(C)C(F)F)=O)C2)cnc2nccn2c1 c1(CNC(C2(C)CN(C(=O)CCC(F)(F)F)C2)=O)ccc2c(c1)CCO2 Cc1ccccc1CC(=O)NC(C)(C)CNC(C1CCC(=O)C1)=O N1(C(C(COC(C)=O)C)=O)C2CCC1CN(C(=O)C(O)c1ccco1)CC2 c1(C(N2CCCC(CN(C(c3ccc(C)s3)=O)C)C2)=O)ccc(S(C)(=O)=O)[nH]1 N1(C(CN(C(=O)OC)C)=O)CCCC(CC(=O)NC2(C)CS(=O)(=O)C2)C1 C1(NC(C(C)CC#N)=O)CN(C(c2ccon2)=O)CCC1(C)C C1(CNC(c2ccccn2)=O)CC2COCC2N1C(=O)COC1CC1(F)F n1(CC(=O)N(C2CCN(C(c3n[nH]cc3Cl)=O)C2)CC)nc(C)n(C)c1=O CC(C)(C(=O)NC1CN(C(c2ccc(S(C)(=O)=O)[nH]2)=O)C2CC12)S(=O)(=O)C1CC1 c1(C(N2CC(C(=O)NC(c3ccno3)C)OCC2)=O)cc2cnccc2[nH]1 N1(C(C2C(CC)C2)=O)Cc2ccccc2C(NC(c2ccoc2Cl)=O)C1 c1(NC(C2CN(C(=O)OC(C)(C)C)C3C2C3)=O)nc2c(s1)CN(C(N)=O)CC2 Cc1cccc(OCCC(=O)NC(C)CC(C)NC(c2cc(F)c[nH]2)=O)c1C c1(NC(C2C(NC(C3CCC(O)C3)=O)CC2)=O)ccc2cccnc2c1 c1(C(=O)NC(C(=O)NCc2cc(C)sc2)CCOCCO)cnc(O)c(C)c1 c1(NC(C2N(Cc3ccc(C)c(C)c3)CCSC2)=O)cc2c[nH]nc2cc1Br N1(C(=O)C=CCBr)CCCC1C1CCN(C(C2CCN(C(=O)C(F)(F)F)C2)=O)C1 Cn1cc(C=CC(=O)NC(CNC(C2(C)CCC(=O)C2)=O)C2CC2)c(=O)n(C)c1=O N1(C(CC(C)CF)=O)CC2(C)CN(C(c3nc(Br)cnc3N)=O)CC2(C)C1 CC1(C)CN(C(c2cc(Br)sn2)=O)CCC1NC(=O)CCC1CCOC1 C1(CNC2CCCC(C=C)C2)CCCc2ccccc2C1 C1(CCC(=O)NCC(=O)NCCC)CCCN1C(=O)C(C)CC c1(OC)nc(OC)nc(N2CCCOC(CNC(C3CNC(=O)N3)=O)C2)n1 N1(C(Cc2nccc(C)c2)=O)C(CC(=O)Nc2cccc(F)c2F)C2CCCC12 N1(C(c2cc(F)cc(F)c2)=O)CC(F)(F)CC1CCO N1(CC)N=C(C(=O)NC2CCCC(NC(C3OCCN(C)C3=O)=O)C2)CCC1=O N1(C(C2CCN(CC)C2)=O)CC2CCN(C(c3cscn3)=O)CC(C2)C1 C(CN=c1nc(N2CCC(O)CC(C)C2)c2c([nH]1)COC2)C1CC(OC)C1 c1(CC)oc(C(=O)NC(C)CCNC(c2cccc(OC(F)F)c2)=O)cc1C Cc1nc2c(o1)CCCC2CC(=O)N1CCC(CNC(c2ccc(C#N)o2)=O)C1 C1(C(=O)NCc2cccc(CNC(c3cc(Cl)no3)=O)c2)CCC2(CCCC2)C1 c1(OC)ccc(CNC(C23CC2CN(Cc2c(O)cccc2Cl)C3)=O)c(C)c1OC c1(CC(=O)NC2CC(CC(=O)NC3(C(=O)NC)CC3)C2(C)C)ccc2c(c1)CC2 C1(NC(C(C)=CC2CC2)=O)CC2CCC1C(NC(c1ccc(C#N)c(C)c1)=O)C2 Cc1nc(O)nc(C)c1CCC(=O)NC1CCCC(NC(c2ccsc2C)=O)C1 C1(C(=O)NCc2ccc(C#N)cc2)C2CC(O)C(C2)N1C(C12CC1CNC2=O)=O CC(O)C(C(=O)N1CCC(CCNC(=O)CCSc2nccn2C)C1)N(C)C C1(CC)C(NC(=O)C(Br)=C(C)C)CCN1C(C1C2CN(C)CC12)=O N1(C(C(C2CCOC2)OC)=O)C2CCCC1CN(C(=O)COC1CCCC1)CC2 Cc1cc(C(=O)NCC(c2ccccc2)NC(=O)CC(C)C(F)F)c2c(c1)CCO2 C1(NC(CN(CCOC)C)=O)CC2CC1CN(C(=O)CCCn1ccnn1)C2 c1(C(c2nnnn2C2CC2)NC2CC(C(C)(C)C)C2)ccccc1C(F)F Cc1cnccc1CCNC(=O)CCOCCN(C(=O)C=Cc1ccco1)C c1(C(=O)NC2CC(O)(CNC(c3c(C(C)C)cco3)=O)C2)cc(F)cc(N)c1F c1(NC(CC2CC(C)N(C(=O)Cn3[nH]cnc3=N)C2)=O)ccc2nncn2c1 N1(C(C(Cc2c(C)nc[nH]2)O)=O)CC2C(CN(C)C(c3cc(N)ccn3)=O)C2C1 c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)COC2)ccc([N+](=O)[O-])c(Cl)c1 C1(C#N)(C(N2CC(NC(C(CC)n3ccc(C4CC4)n3)=O)C2)=O)CCOCC1 c1(NCCCOCCNC(C(C)NC(=O)NC)=O)ccc(C)c2[nH]c(C)cc12 c1(C(N2CC3CC(CNC(C4(OC)CC4)=O)C3C2)=O)c(O)nnc2c1COCC2 C=CC(C)(CC)C(=O)NC1C2CCC1N(C(=O)C(c1ccccc1)N(C)C)C2 N1(C(C2C(COC)C2)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 CN1CCC(N2CCC(O)(CNC(=O)Cc3nc(C4CC4)nn3C)C2)C1=O C(=O)(C(C)(COC)CC)NC1(C(=O)NC(CCC)C2CC2)CCSC1 N1(C(CCC#C)=O)CC(NC(c2cc(C3CC3)oc2C)=O)C(C2CC2)C1 C1(C2CCN(C(c3cnc4c(c3)NCC(=O)N4)=O)CC2)(C(=O)OC)CCC1 C(=O)(CC1=CCCC1)N1C(CNC(C2CC(CO)C(O)C2)=O)CC1 c1(C(=O)NC(C2CCN(C(c3ccncc3F)=O)CC2)C)ccn(C)c(=O)c1 N1(C(C(CCOCC)NC(=O)CC=CC(C)(C)C)=O)CCOCC(OC)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCCCC1CCC(=O)NCC(F)(F)Cl C(c1ccc(C)cc1)=CC(=O)NCc1c(C(N(CC(CC)(O)CC)C)=O)con1 N#CC1CCC(NC(C2CN(C(=O)COCC3CCOC3)C2)=O)CC1 N1(C(c2[nH]ccc(=N)n2)=O)CC2(CCOCC2)CC1CNC(C1CCCCS1)=O C1(NC(C2CN(CC(C)C)C2)=O)CN(C(c2cncc(C)n2)=O)CC(C)(C)C1 c1(C(N(CCNC(C2CCC2C2CCCO2)=O)CC)=O)ccc(C)c(C)c1 C12(NC(c3c(C)ncnc3O)=O)CCCC1N(C(=O)CCC(C)(F)F)CC2 Cc1nc2ccc(C(=O)NCC(C)N(C(=O)CC(C)(F)F)C)cc2o1 Nc1cccc(F)c1NC(C1CC(n2cc(C3CCOC3)nn2)C1)=O c1(OC)ccc(C(N2C(C(=O)N=c3cc(CCO)[nH][nH]3)CC3CC23)=O)c(C#N)c1 c1(C(=O)NCCCNC(c2ccc(NC)cn2)=O)coc2c1C(O)CCC2 N1(C(C(C)OCC)=O)CCC(NC(c2c[nH]nc2-c2ccsc2)=O)CC(C)(C)C1 c1(OC)cc(OC)c(NC(C2(C)CCN(Cc3cccc(C#N)c3)C2)=O)cn1 C1(CC=C)(NC(c2cnn(CC3CC3)c2)=O)CN(C(c2nonc2N)=O)C1 C(=O)(CCCCC(F)(F)F)NC12N(C(C(C)(C)C3CC3)=O)CC(CO)(C1)C2 c1(C(N2CCC(N(C(=O)C=CCF)CC)C2)=O)ccc(Cl)c(Cl)c1OC Cc1ccc(C(=O)NCC2CC(C)N(C(c3ccc(C(N)=O)s3)=O)C2)cc1C#N Cc1cccc(C(=O)NC(C)CNC(c2ncc(Cl)cc2O)=O)c1Br N1(C(C2CN(CC)C(=O)N2)=O)CCCC(CO)(NC(=O)CCc2cc(Cl)no2)C1 C(c1ccc(C)nc1)=CC(=O)NC(CNC(c1cncc(COC)c1)=O)(C)C N1(c2nccc(OCCC)n2)CCC2C(CCCN2C(C2COCCO2)=O)C1 C1(CC(=O)N(C2CCN(C(=O)CC3(O)CCOC3)C2)CC)CC=CCC1 N1(C(c2c(COCC(=O)Nc3ccsc3)c[nH]n2)=O)CC2(CCCC2)C1 N1(C(CCC)=O)CCC2CCN(C(=O)C(c3ccc(F)cc3)N(C)C)CC12 N1(C(Cn2ccc(C)cc2=O)=O)CCCN(C(C2C=CCCC2)=O)C(C)C1 c1(CC)oc2ccccc2c1C(=O)NC1CC1CNC(=O)C(C1CCOCC1)F CC1C=C(C(=O)NCCOC2CN(C(=O)COc3cccc(F)c3F)C2)CC1 C(=O)(C1=COCCC1)N1CCCC(N(C)C(C2(C)CC=CC2)=O)C1 C(CC(C)(C)C(=O)NCC1CC(F)(F)CN1C(=O)C(C)Sc1ccccn1)SC NC(CC(F)F)C(=O)NCc1sccc1I N12C(C3CCCC13)CC(=O)N(CCCCC(F)(F)F)C(C)(C)c1c(C)oc(c1)C2=O.C(C)C.CO c1(NC(C2=CCC(NC(c3c(C)cn(C)c3)=O)C2)=O)cc(C)c(O)c(C)c1 C(=O)(CC(O)CNC(C1CC1Cl)=O)Nc1cn(CC=C)nc1 c1(NC(C(C)OCCC#C)=O)cccc(NC(C)CCc2ccc(Br)cc2)c1 c1(C(=O)NC2(C)CCN(C(Cc3nc(CC)sc3)=O)C2)nc(C)n(C)c1C CC1CC(C(=O)NOCC(C)(C)O)N(C(c2ccc(CCN(C)C)cc2)=O)C1 C1(CNC(CC2(CCOCC=C)CCC2)=O)CCC(C(=O)CC2(N(C)C)CCC2)C1 CCC(C)(CO)C(=O)N1CCN(C2CN(C(c3cnn(CC4CC4)c3)=O)C2)CC1 c1(NC(=O)Nc2c(C)nc(F)cc2)ccc(S(=O)(=O)NCc2nncn2C)cc1 C(C1CCCN1C(=O)CCCn1cccc1)=CC(=O)NC1C(C)(C)CC1 N1(C(CCCSC)=O)CC(CNC(c2cccnc2C2CC2)=O)C(C(F)(F)F)C1 CC(C)(C)CC(O)CC(=O)N1CC(O)(CCNC(C2(CO)CCCC2)=O)C1 Cc1cc(C(N2CC(C(=O)NC3CCNC(=O)CC3)CC2(C)C)=O)cc(F)c1 c1(C(C)(C)C)cccc(-c2cn(CC(F)(F)CNC(=O)CC#N)nn2)c1 CC1CC2CN(C(C34CC5CC3C4C5)=O)CC2N1C(C1C2CC(F)(F)CC12)=O N1(C(CC(=O)OCC)=O)CC2(CC(NC(c3ccc(CO)cc3)=O)C2)C1 Cc1cc(C(=O)NC2(CNC(C3(C4CCCO4)CCC3)=O)CC2)c2[nH]cnc2c1 c1(C(=O)OC)ccc(CNC2CCCC2C(C)(C)C)cc1OC(F)F c1(N2CCC3(CC(OC)C3)C2)nc(=NCC(C)S(C)(=O)=O)[nH]c2ccccc12 N1(C(c2n(COC)ncc2C)C(=O)NC2CCCC2)CC2CC(C1)N2CC(F)F c1(CC(=O)NC2CCC(CNC(C(C)(Cl)Cl)=O)C2)cccnc1Cl C#Cc1ccc(C(N2CCN(C(=O)Cc3cncc(C)c3)CC(O)C2)=O)cc1F C1(C(N(CCC(N)=O)C)=O)CC2C=CC1N(C(C1SCCS1)=O)C2 O=C(N1NC2CC1C(O)C2O)c1ccccc1.C1(N)CNC1 CCCC(C)(C)CNC(=O)C(C)(CO)NC(c1cncnc1C)=O O=S(=O)(c1ccc2[nH]c(=NCc3ccc(Cl)cn3)sc2c1)NCCCOC1CC1 N1(C(CCCOC(C)C)=O)CC2(C1)CN(C(c1c(N)cc(Cl)cc1F)=O)CCO2 CC(CC(=O)N(CCCCCCNC(c1ccnn1CC(F)(F)F)=O)C)C(F)F N1(C(C(C)C)=O)CC2CN(Cc3ccccc3CN)CC2C1 N1(C(=O)NCC2(CC(C)C)CCC2)CCC2CSCC2C1.NC C1(C)(OC)CCCN(C(=O)COc2cccnc2)CC1.C12CCN(C1)C2=O C(C(C)(COC)C(=O)N1CCC(COC)(NC(=O)CC2CC(C)=NO2)C1)OC c1(NCCC2(OCC)CCOC2)[nH]c(=NCc2cnn(C)c2)nc2ncn(C)c12 c1(CC)ncoc1C(=O)NCC(n1cc(C(C)CN2CCCC2)nn1)C C1(C)(C2(C(=O)NCc3cn(CC)nc3)CC2)CCCN1C(c1cc(Cl)n[nH]1)=O C1(NC(CC2CC(CC)C2)=O)CCC2(CCCN(C(=O)C(C)(F)F)C2)C1 C1(C(N2CCOC(CN(C(=O)CN(C)C3CC3)C)C2)=O)(CC)CCC(F)(F)CC1 C(=O)(CCCC(=O)NC)NC1C(CC)CN(C(=O)CSC(C)C)C1 C(CC(=O)NC1CCCCC1F)(C(F)F)NC c1(CNC(C2COCC2n2cc(-c3ccccn3)nn2)=O)ccc2[nH]ccc2c1 C(C)(C)(CC(=O)NCC(c1ccccc1)N(C)C(c1csc(C(N)=O)n1)=O)OC CC1=NNC(=O)C1CCC(=O)NCC1CCC1NC(=O)Cc1nn(C)cc1Cl C1(NC(c2ccnn2CC(F)(F)F)=O)CCN(C(=O)C2=NOCC2)C(C2CC2)C1 c1(OC)nc(C)c(C(N2CCC(C)(CCNC(c3ccc(O)cn3)=O)C2)=O)s1 N1(C(C2CC(C)OCC2)=O)CC2(CCCC2NC(=O)CCc2cnoc2)C1 Cc1cc(Br)ccc1-n1cc(C(C(C)C)NC(=O)C(O)c2ccco2)nn1 C1(CN(C(=O)CC2CCCCC2)C)CCCCN1C(c1cc(C(F)(F)F)no1)=O C(=O)(C(C(C)(C)C)NC(c1ccc(Cl)cc1Br)=O)NC1(C#C)CC1 CCCC(CCCNC(C12CC(C#N)(C1)C2)=O)NC(=O)COc1cccc(F)c1 c1(OC)cc(OC)cc(CC(=O)N(CCCNC(c2c(CO)nnn2C)=O)C)c1 C1(NC(C2CC2c2ccc(F)cc2F)=O)CCCN(C(C2CCOC2)=O)CC1 C(=O)(C(C1CCC1C(F)(F)F)N(C(C)CC1CCCC1)C)NCC(=C)C C(=O)(C(C)(O)C1CCC1)N(CCC)CCNC(=O)CC1CC(=O)C1 N1(C(C=NOC)=O)CCC2C(CCCN2C(c2ccc(F)c3cccnc23)=O)C1 C1(NC(C(=O)NCC(F)F)=O)CCCCCN(C(c2ccc(F)c(Cl)c2)=O)C1 C1(NC(C2C3CNC(=O)C32)=O)CN(C(=O)Cc2ccccc2Cl)CC12CCC2 S(=O)(=O)(c1ccc(S(=O)(=O)NC2CCC2)c(Br)c1)N(CC(C)(C)CCCO)C C1(C(=O)NCC2OCCN(C(C)C(=O)Nc3ccccc3)C2)CC12CCOCC2 C(=O)(C(C)(C)C(N)=O)NCCC(C)NC(C(CSC)OC)=O C1(CNC(=O)CN2CCCC2)CCCC(CNC(c2csnn2)=O)C1 C#CCC(C)(C(=O)N1CC(NC(=O)NC)C1)NC(C1CC2C(C1)C2(C)C)=O N1(C(Cc2nc(C(C)C)on2)=O)CCN(C(c2ccccc2C#N)=O)C2(CC2)C1 N1(C(c2c(CC)n[nH]c2)=O)CC2CCCC2(NC(C2CC23CC3)=O)C1 C(CC(=O)NCC(C)(C(C)C)NC(C1CC(C(C)(C)C)=NO1)=O)(C(F)(F)F)OC C1(NC(C2CC(C(C)C)C2)=O)COC2(CCN(C(c3c[nH]ccc3=O)=O)CC2)C1 N1(C(c2cc(OC)n[nH]2)=O)CCN(C(c2ccc(CO)nc2)=O)C(CN(C)C)C1 c1(C(N2CCC(NC(COCCCOC)=O)C2)=O)cc2c(Cl)nccc2o1 c1(NC(=O)NC(C)Cc2nn[nH]n2)nccc(N(C)CCOC)n1.C(C)(C)(C)O C1(N(C(C=CCCC)=O)CCF)CCCN(C(c2c(C)coc2C(C)C)=O)C1 CCC(CC(=O)NCC(C)(C)CNC(C1CCN1C1CCCC1)=O)SC C1(CN2CCC(c3ccc(C#C)cc3)CC2)CCc2ccccc2NC1=O C(=O)(C1=C(Cl)CCCC1)N1CC(CCCCNC(C(C)NS(C)(=O)=O)=O)C1 CN1C(=O)Cc2ccc(C(=O)NCC(O)CN(C(=O)C(O)C(F)F)C)cc21 C1(C(N2C(C)C(C(=O)N(C)CCN(C)CCO)CC2)=O)CCN(C)C(=O)C1 C1(NC(c2n(C3(CC)CC3)nnn2)C2CCC2)CCc2n[nH]cc2C1 n1(C(COC)C)nc(-c2ccccc2Br)nc1-c1ccc(Cl)cn1 C1(C(N(c2ccc(OC)cc2)c2ccc(Br)cc2)=O)CC12CCCNC2 c1(C(=O)NC(CC(C)NC(c2c(C)nn(C)c(=O)c2)=O)C)ccc(Cl)c(Cl)c1O c1(CC)ccc(Cl)c(C(=O)NCCCC(C)NC(C2(C)CNC(=O)C2)=O)c1 C(CCCC(=O)O)CN(C(CCCc1c(C(=O)OC)scc1)=O)C12CC(C1)C2 N1(C(CCC(C(C)C)NC(=O)CC(O)CC(C)(C)C)=O)CC2C3C=CC(C3)C2C1 C(C(=O)N(CC(O)CNC(=O)CCC1(C)CC1)C)(C(C)C)n1ncc(C)c1 C1(NC(CCC2(C)CC2)=O)CN(C(c2cnn(C)c2C(F)F)=O)CC2CC12 c1(C(=O)NCCCNC(C(C=C=C)C)=O)c(F)c(F)cc(F)c1F c1(OC)ccc(C(N2CCC2C(=O)Nc2cc(C(N)=O)nc(Cl)c2)=O)c(Cl)n1 CC(C)C(CN(C)C)NC(=O)CCc1nc(-c2ccco2)n[nH]1 c1(C(=O)NC(CNC(C2(C(=O)OC)CC2)=O)CO)cc(OC)c(OC)c(Cl)c1 c1(CNc2nccc(CNC(=O)CC3CCC(=O)N3)c2)ccc2c(c1)CNC2=O N1(C(c2n(C)ncc2Cl)=O)CCCN(C(=O)CC2CCCNC(=O)C2)C(CO)C1 c12c(cnn1C)NC2=O.c1(NC(C2CC3(CC3)C2)=O)ccc(COC)cc1 N1(C(c2ccc(C)s2)=O)CC2CCC(N=c3nc(-c4ccccc4)[nH]s3)C2C1 N1(C(CC=C)=O)CCN(C(c2cc(C(=O)OC)no2)=O)C(CO)C1 C1(C(=O)NC2CC(CNC(c3ccc(N4CCCC4)nc3)=O)C2)CCC2(CCC2)O1 N1(C(c2c(C)noc2C)=O)CCC(C)(C)C(C(=O)Nc2cncc(CO)c2)C1 Cc1nc(C(=O)NC2CN(C(=O)C(C)O)CC2c2cn(C)nn2)c(C(F)(F)F)[nH]1 CC1=C(C(=O)NC(C)CCNC(=O)C(O)CC(N)=O)Cn2nnnc2N1C c1(C(=O)NC2CC(C)(NC(c3cnc(CCC)s3)=O)C2)cncc(C)n1 N1(C(C(C=C)OC)=O)CCN(C(=O)Cn2nnc(C)n2)C(c2ncc[nH]2)C1 N1(C(C(CCSC)O)=O)CCC(NC(=O)C2=C(Cl)CCC2)C(O)C1 CCC(C)C(C(=O)N1CC2CC1C2C(=O)OC)NC(c1cc(F)cnc1O)=O c1(C(N2CC(CNC(C3CCSC3)=O)C(O)C2)=O)cc2cnccc2[nH]1 C1(C#CC(=O)NC(C)CCCNC(c2cnc(C3CCC3)nc2O)=O)(CC)CC1 CN1C2CCC1CC(C(=O)NCC1(F)CCC(NC(c3ccsc3)=O)C1)C2 N1(C(C(C=CCCC)O)=O)CCN(C(=O)COc2cnccc2C(F)(F)F)CC1 c1(CC)cc(C(=O)N(CC(C)C(=O)NCCC2CCSC2)C)nn1C O=C(NNc1cccc(CCN2CCCC2=O)n1)c1cc(I)ccc1C(F)(F)F CC1(C)CN(C(=O)Cc2ccoc2)CCN(C(C2(C#N)C(C#N)C2(C)C)=O)C1 c1(CC)nn(C)c(CC(=O)NCC2CC(C)(C)CN2c2cnc(C)cn2)c1Br Cc1sccc1CC(=O)NC(c1ccccc1)C1CCCN1C(=O)C(C)(F)F c1(NC2(C(=O)NCC3(NC(c4cc(Br)c[nH]4)=O)CCC3)CC2)ccccc1 CC1CN(C(c2cc(C(F)(F)F)ccn2)=O)CC1CNC(c1cncc(O)c1)=O C1(C(N(C(C)C(=O)NCC(C)(C)O)CCC)=O)CCCC1C C1(CNC(C2CN(C(C)=O)C2)=O)CC2CN(C(c3cnc(O)o3)=O)CC12 c1(OC)ccc(F)c(C(=O)N(CCCNC(C2CCC3CC23)=O)CCO)c1 C(=O)(CCC(=O)c1cccc(Br)c1)N(C)Cc1onc(CC)n1 Cc1c(F)cc(C(=O)NNC(=O)c2ccc(Cl)cc2)c(C)c1N c1(CC)nccn1C(=O)NC1CCOC1CC(C)C C1(C2(C(N(CC(C3CC3)NC(C3(n4nccn4)CC3)=O)C)=O)CC2)(CO)CCC1 C1(F)(CNC(C2CC2C2CC2)=O)CCN(C(c2cn(C3CC3)cn2)=O)C1 c1(C(C)NCCC2CCC3CC23)cc(Br)ccc1[N+](=O)[O-] c1(CC=C(C)C)ccccc1CNC(=O)C(C(C)C1CC1)N(C)CCN(C)C.CO NC1CC2CN(C(c3ccccc3-c3cccnc3)=O)CCN2C1=O CC(C)(C)C(CNC(=O)COc1ccccc1C(F)F)NC(C1C2CCCC12)=O c1(-c2n(CCC=C)c(N3CC(C)SC(C)C3)nn2)cnc2[nH]ncc2c1 C1(NC(c2n(C)c(S)nc2)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)C12CCC2 N1(C(C23CC2CN(Cc2c(F)ccc(O)c2F)C3)=O)CCC(O)C(F)(F)C1 N1(Cc2n(C)ncn2)CCC(NC(c2ccc(C(N)=O)[nH]2)=O)C(O)C1 C1(C(=O)NCc2oc(C(=O)NCCOCC(=O)OC)c(C)n2)CCC(O)CN1C c1(C(=O)NCCCCC(C)NC(=O)C(C)(C)F)cc2ncccc2cc1Cl C12(CNC(CC3(NC(C(CC=C)OC)=O)CCC3)=O)CCC(C1)C(=O)N2 N#CC1CN(C(C2(CNC(c3ccc(CO)cc3)=O)CC2)=O)CCO1 C(=O)(C1=C(C)OCCS1)N1C(CN(C(C(CCC)O)=O)C)CCC1 CCCC(CCC)C(=O)NCC(O)CNC(c1ccc(Br)nc1OC)=O C1(CC(N2CC(OC)C(NC(C3(O)CCCCC3)=O)C2)=O)OCCCC1(C)C N1(C(c2c(C)con2)=O)CC2CCC(C1)N2C(c1ccn2c1CCCC2)=O n1(CCC)cc(NC(C2CC(n3cc(C4(COC)CC4)nn3)C2)=O)cn1 C=CCC(C(=O)N(C(C(=O)NC(c1nccs1)C)C1CC1)C)C(C)C CC1C2CN(C(C3(C)CC(NC(=O)OC(C)(C)C)C3)=O)CC12 N1(C(CCC(=C)C)=O)CC(C)CN(C(=O)C(c2ccccc2)OCC)CC1C N1(C(c2nccc(C)c2)=O)CCN(C(=O)CN2CCCC2=O)CC(C)(F)C1 c1(OC)cc(C)nc(NC(C2CC23CN(Cc2c(Cl)ccnc2Br)C3)=O)n1 N1(C(C=CC)=O)CC(NC(=O)CNc2ccccc2C)C(c2nccn2C)C1 CC1CCC(NC(C2(C)CCCOC2)=O)CN1c1ccc(C#N)nn1 c1(C(=O)NC(C2CCCC2)CNC(C(CC2CC2)OC)=O)ccc(Cl)nc1N c1(SC2CC2)cc(C(N2CCC(NC(CCC3CCN(C)C3)=O)C2)=O)ccn1 C(=O)(CC(C)(F)F)NC(C1CCN(C(=O)C(C2COC(C)(C)O2)O)CC1)C n1(CC)c(C)cc(C(=O)NC(C2CCCN2C(=O)C=CCCC(C)C)(C)C)c1C N=c1[nH]c2ccc(CN3CCC(C(=O)Nc4cccc5occc45)C3)cc2s1 C=Cc1ccc(C(=O)N(CCCNC(=O)CCc2ccc(O)c(Cl)c2)C)cc1 C1(OCCC)CN(C(=O)CCOCC)CC1CNC(C1CC(=O)C1CSC)=O c1(C(=O)NCCCN(C(=O)CCc2cscn2)C)cccc(S(C)=O)c1 C(CCOCCO)(C(=O)N(C)Cc1cncnc1)NC(C(C1CCC(=O)N1)C)=O N1(C(C2N(C(CCCC)=O)C3C(C2)C3)=O)CCC(C2CCOC2)C1 Cc1cc(C)c(C(N2CCSCC2CCNC(=O)CC2CCCOC2)=O)o1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(CCCNC(C(C(C)C)F)=O)CC1 N1(C(c2c(CC)oc(C)c2)=O)CC(C(=O)N(CC)CC2CCCO2)CC1(C)C n1(CC(=O)N(CCCNC(COc2cc(C)on2)=O)C)cc2ccccc2n1 C12(C)COCCN(C1)C(=O)NC2.S(=O)(=O)(c1ccc(C(=O)OC(C)(C)C)s1)N(C)C c1(CCOC)ccc2c(c1)OCC2C(=O)NC(=O)C(N1CC2CCC1CC2)=O C(c1ccsc1)=CC(=O)NC(CC1CC1)C(=O)NCc1ncsn1 C(=O)(CS(=O)(=O)N(C)C)N(C)CCNC(c1ocnc1C(F)F)=O C1(OC)(CNC(=O)CN(CC(C)(C)C)C)CCN(C(C2(O)CC2(C)C)=O)C1 C1(NC(CNC(C)=O)=O)CCN(C(c2cc(C#N)n(C)n2)=O)C12CC2 Cc1ccc(CC(C)C(=O)NCC(C)NC(=O)Cc2c(Br)cnn2C)cc1 C1(NC(CC2(OC)CC2)=O)CCCN(C(C23CC4CC2C3C4O)=O)CC1 Cc1c(C(=O)NCC(O)CCNC(=O)C2=C(Cl)CC2)c[nH]c2nccc1-2 N1(C(CC(C=C)(C)C)=O)CCCN(C(c2cccc(OC)c2C)=O)CC1C C1(CC)(NC(c2ccc(C3CCOC3)cc2)=O)CCCN(C(=O)CCC2CC2)C1 c1(N(C2CCN(C3CC3)CC2)C)ccc(C2CC2)c(C#N)n1 C=CCC(CO)NC(c1occc1CNC(=O)C(n1nccc1C)C)=O C1(NC(c2cc(C(C)C)on2)=O)CCCC12CN(C(C1(C3CCCO3)CC1)=O)C2 Cn1ncc2cc(C(=O)NCC3CCCC3NC(=O)Cc3ccsc3)cnc12 CCCC(CC)CCC(=O)NC(C(=O)NCC(C(C)C)C(C)C)c1ccoc1 c1(C(N2CCC=C(C(=O)NC(C)CO)C2)=O)ccnc2c(O)cccc12 Cc1ccc(F)cc1C(=O)NC1CCCC(C(N2CC3(CC3)C2)=O)C1 N1(S(CC)(=O)=O)CCN(Cc2c(C)cc(OC)cc2C)CC1C#N C1(C(N2CCCN(C(CCC(C)OCC)=O)CC2)=O)CC12CCC(F)(F)CC2 C(=O)(C(CNC(c1coc(C2CC2)n1)=O)C(C)(C)C)N(c1ccccc1)CC Cc1cn2cc(N(C3CCNCC34CC4)C(=O)CN(C)C)ccc2n1 c1(CNC(C2N(C(CSCC)=O)CC=C2)=O)ccnc(O)c1 c1(C(N2C(CCNC(c3n(C)nnc3)=O)CSCC2)=O)cccc2[nH]ccc12 C1(C(N2CCCCC2CCN(C)C)C(=O)NCC(C)C)C(F)(F)C12CCC2 c1(C(=O)NCCC(C)N(C(c2ncn(CC)n2)=O)C)nc(C)ccc1O N1(CC(=O)NCCC(=O)N(CC)CC)CC2CC3CC(C2)CC1C3 n1(C(CC)C)nccc1C(=O)N(C(C)CNC(c1nncn1C1CC1)=O)C c1(NCc2c(NC(C(C)NC(=O)OC(C)(C)C)=O)cccc2)ccc(Cl)c(Cl)c1 Cn1cnc2c1C(C(=O)NC1CC3C1CCN3C(=O)Cc1cccs1)CC(=O)N2 C1(NC(c2cccc(OCC(C)C)c2)=O)CC2CN(C(c3n[nH]cc3Cl)=O)CC12 c12ccc(cc1)[nH]c2=O.N1(C(CC2(C)CC2)=O)CC(N(C(=O)C=NO)C2CC2)C(O)C1 CCC(CC(=O)NCC(Cc1ccccc1)NC(=O)C=C(C)C(C)C)OC CC(C)C(CC(=O)NCC(CO)C1CC1)NC(c1cnn(C2CC2)c1)=O c1(C(=O)NC(CNC(C(C(C)OC)O)=O)C(C)C)nc(C)ccc1O c1(CC)cc(C(=O)NC2CC23CC(NC(=O)CCCC2CC2)C3)cn(C)c1=O C1(NC(C)=O)CCC(C(N2CC(NC(c3nnc(C(F)F)s3)=O)C(C)C2)=O)CC1 CC(C)CCC(F)C(=O)N1CCC(CF)(NC(=O)CC(C)n2ccnc2)C1 N1(Cc2cnc(C)s2)CCCc2ccc(NC(c3cc(Cl)ccc3O)=O)cc2C1 C1(NC(C2CCCC(OC)C2)=O)CC(F)CN(C(=O)C(C)(CO)NC(C)=O)C1 c1(OC(N(C)CC2CCN(C(=O)Cc3ccnc(F)c3)C2)=O)cccc(C(N)=O)c1 N1(Cc2c(Br)cn(C)n2)CCC(=O)N(CCSCc2ccccc2)C1=O CC1CN(C(C2(Br)CC2)=O)CC2(CCN(C(C3C4CCC3CC4)=O)C2)O1 N1(C(C2CC(CCC)C2)=O)CC(C2CCN(C(=O)CC3CCOC3C)CC2)C1 C1(C(N2CC(CC)(OC)C2)=O)CC(C)CN1C(C1CCC(CO)CC1)=O.C1CC1 c1(OC)cc(Cl)ccc1C(=O)NC1CN(C(=O)CC2CCCCC2O)CC12CC2 C12(NC(C(C)n3cccc3)=O)CC(CNC(=O)CCNc3ccccn3)(C1)C2 N1(C(C2C(C(=O)O)CC2)=O)CCNc2ccc(F)cc21 C1(C)(CC)C=C(C(=O)OC)C1.C(C(F)(F)C(F)F)ONC(c1ccc(CNC=O)[nH]1)=O C1(CNC(CSCCC(C)C)=O)CCCCN(C(=O)CC2(O)CCOC2)C1 CCCCC(CC)C(=O)N1CCCC(CC(=O)NC2CCCC(C)(C)C2)C1 c1(CC)cc(C(N2C(C(=O)NC3CSC(C)C3)CCC2C2CC2)=O)c(C)o1 C1(CC)CC(C(=O)NCC(C)C(=O)OC)CCN1C(=O)C(C)c1cc[nH]n1 c1(C(=O)OC)cc(C(N2CCC(NC(c3cccc(C4CC4)c3)=O)C2)=O)ccn1 C(CCCCC(=O)N1CCCCC1CO)NC(CC1CCC(=O)N1)=O C1(C(=O)NC(C2CCCN2C(c2ccnc(O)c2)=O)(C)C)CC2CCC1CC2 C12(NC(Cc3c(C)non3)=O)CC3CC(C1)CC(NC(C14CC(C)C1C4)=O)(C3)C2 N1(C(C(C)C(F)F)=O)CC2(C1)CN(C(C1CCOCC1)=O)CC(C)(C)O2 N1(C(C2C(C)C2)=O)CCC(N2CCC(NC(C3CC4CC4C3)=O)C2)CC1 C1(CC(N2CC(NC(C3CCC=CO3)=O)C2)=O)CN2CCN1CC2 c1(C(N2CCC(C(=O)Nc3ccc(C)nc3Br)CC2)=O)cc(F)c(CO)cc1F C(=O)(C(C)(C(C)C)NC(=O)C(C(C)C)NC(=O)NC)N(CCCC)CC C1(C(N(CC(C)C)C(C)C)=O)CN(C(c2ccc(Cl)cn2)=O)CC(C)(C)C1 c1(C(=O)NCC2OCCN(C(C(CC#C)O)=O)C2)cc(C)cc(Cl)c1 N1(C(C(=O)N(C)C)=O)CCN(C(C2COC3(CCC3)C2)=O)C2CCCCC12 N1(C(CCC)=O)CCC2(CC2)CC1C(N1CCCOCC1C)=O C1(C(=O)NCc2ccc(CC)o2)CCC2CC1CO2.C12(CCCO1)C(=O)N(C)C2 N1(C(C(=O)NCC)=O)CCC2CCC(NC(=O)C(F)C(F)(F)F)C1C2 c1(CNC(=O)NC(C2CCCO2)COC)ccccc1C#Cc1ccccc1 c1(C(=O)NC(C2CN(C(c3cccnc3C3CC3)=O)C2)C)cc2c([nH]1)CCCC2 c1(N2CCC3(c4nnc(C)n4C)C(C2)C3)nc2cc[nH]c2c(=NC(C)C)[nH]1 n1(CC)ncc(C(=O)NCCC2CCC(NC(=O)CCN3CCCC3=O)C2)c1C N1(C(c2cnc(C)o2)=O)CC23CCCC2(C1)CN(C(=O)CC(C)C(F)(F)F)C3 n1(CC)cnc(NC(=O)N(CC(C)(O)C2CC2)C(C)C)c1 C1(C(=O)N(C(C)CC(N)=O)C)(CC)CCN(C(c2ccoc2)=O)C1 C#CCCCC(=O)NCC1CC(C(F)(F)F)CN1C(C1CC(Cl)(Cl)C1)=O c1(C(N2CCC(CCNC(=O)C(F)C3CCC3)C2)=O)cc2cc(Cl)ccn2n1 C1(N(C(CCC)=O)C)CCCN(C(c2ccc(C(C)(F)F)nc2O)=O)CC1 C(=O)(C(C)CS(C)(=O)=O)NCCC(CNC(C1(C(=O)NC)CCC1)=O)OC N1(C(C(CC)CC)=O)CC(NC(c2ccn(C3CCCC3)n2)=O)CC(O)C1 C(=O)(CC=CC(C)(C)C)NCC1(CC(=O)NC2C(CC)C2)CC1 C1(C(N(C)CC2OCCN(C)C2)=O)CN(C(c2cnc(Cl)n2C)=O)CC12CCC2 c12oc(nc1C#N)[nH]2.N1(C(C(=O)N(C)C)=O)CC(C)(CC(=O)N2CCC2)C1 c1(C(=O)NC2(C)CC(NC(C3CCCN(C)C3)=O)C2)n[nH]c2cccnc12 c1(C(=O)NC(CC)CNC(C2CCCCC(=O)N2)=O)cc(C)ccc1S(N)(=O)=O N1(C(C2CC(C)OCC2)=O)CC2(C1)CN(C(c1cc(C3CC3)on1)=O)CC2CO C1(NC(c2coc(Cl)n2)=O)CCN(C(=O)CSc2nncn2C2CC2)C1 C(=O)(CCC(=O)NCCC1CN(C(=O)C(F)C2CCOC2)C1)c1cn(C)nc1 C1(CNC(CN(C(CCN(C)CC)=O)C2CC2)=O)NC(=O)OC1(C)C c1(C(=O)NCCOC2CN(C(C3(C)C(C)C3)=O)C2)ccnn1C1CCCC1 N1(C(CCC=CC(C)C)=O)CCC(C)C(NC(c2ncsc2C(C)C)=O)C1 CCC(C(=O)NCC1CC(F)(CNC(=O)CC2(OC)CCCC2)C1)C(C)C C(C(=O)NC1C2CN(c3ccnc(C(C)C)n3)CC12)(C(C)C)OCC C(=O)(CCCCNC(N)=O)NC(C(c1ccccc1)NC(CC(=O)NCC)=O)C N1(C(C(CSC)O)=O)CC2CCCC2(CNc2ncncc2Cl)C1 c1(CC(=O)NC2(CO)CN(C(=O)CC3(CO)CC3)C2)cccc(Br)c1F c1(Cc2cn(C3C(C)N(C(c4cc(F)c[nH]4)=O)CC3)nn2)cc2scc(Cl)c2[nH]1 c1(C(N2C(CNC(c3c(Cl)ccc(OC)c3)=O)CCC2)=O)c[nH]nc1S(N)(=O)=O N1(C(C(CC#C)O)=O)CC23CCCC2(C1)CN(C(c1ccnn1CCCC)=O)C3 CC1CCN(C(=O)CC2CCOCC2)C1CNC(C12CC(C1)C2)=O c1(OCC)cc(C(N2CCCN(C(c3ncon3)=O)CC2)=O)ccc1C CCC1=NOC(CC(=O)N(CC(CC)NC(c2cc(COC)cs2)=O)C)C1 C(=O)(C1=C(C#N)CCC1)NC1CC(F)(CNC(COCc2n(C)ncc2)=O)C1 CC(CCC(=O)N1CCCC1CCNC(c1sccc1Cl)=O)N(C)C c1(C(=O)NC2C(CNC(c3c(C)ncs3)=O)CC2)cc2cc(Br)ccc2o1 C1(NC(C2N(C(C)C)C(=O)CC2)=O)CC2CN(c3ncncc3I)CC12 C1(C(c2cscc2Cl)=O)(NC(C2CN(C(=O)NC)C2)=O)CCCC1.C(CN)O Cn1cnnc1CCCNC(C1CC(NC(C2(CCCF)CC2)=O)C1)=O c1(C(=O)NC2CCC2NC(C2CC(C(F)(F)F)C2)=O)c(Cl)cccc1Cl C(=O)(CC(C)(C)C(F)F)N(CC(C)NC(C=Cc1cccc(OC(C)C)c1)=O)C N1(C(C2CC(CNC(c3ccccc3F)=O)C2)=O)CCC(F)(F)CC1 CC1(C)OCCC1C(N1CCCCC1CC(=O)N(C1CC1)CC1CCC1)=O n1(CC)ccc(C(=O)NCC(C)N(c2nnc(C3CC3)o2)C)n1 c1(C(N(CCNC(C2CCC(SCC)C2)=O)C2CC2)=O)sccc1S(=O)(=O)NC c1(C(=O)NC(c2ccc(C)cc2)CNC(C(CCC)O)=O)cc2ccccn2c1 c1(C(N2CCN(C(CC(=O)OC)=O)C3C2C3)=O)cc(Br)c(OC)cc1N C12(NC(C(c3cccc(Cl)c3)C)=O)CC1CN(C(=O)C=Cc1ccn(C)c1)C2 Cc1cccc(C(=O)NCC(C)(C)C(=O)N2CCOC(C3CC3)C2)c1O N1(C(CC(=O)OC)=O)CCCCC(C(=O)N(CCF)C2CC2)C1 C1(C(C2CC(F)(F)C2)C(=O)OC)CN(C(=O)Nc2cncc(O)c2)CCO1 c1(NC(CCCC)CC)ccc(S(=O)(=O)NCC2CC2(C)C)cc1Br CC1CC(NC(=O)CN(CC(C)(C)C)C)CN1C(C1CC(N(C)C)C1)=O c1(SCC(=O)OCC(=O)NCCn2cc(CNCCC)nn2)cccc(F)c1 C(=O)(C1CCCc2nncn21)NCC(CNC(C1=NOC(C)C1C)=O)(C)C CC(C)CCC(=O)C(=O)N(CCC(N1CCC([N+](=O)[O-])CC1)=O)C N1(C(C2C(=C)CC2)=O)CCC(C2CCN(c3ccc4nccnc4n3)CC2)CC1 N1(C(C(C2CC2)OCC)=O)CSCC1C(=O)NOC1CCCC1 C=CCC(CNC(c1c(C)cnnc1O)=O)C(=O)NC(Cn1cncn1)CC C1(CO)CC2CCC(C1)N2C(C(=O)NCc1c(C)n(C)nc1)C1CC1CC(C)C C=CC(CC)CC(=O)NCC(=C)CCNC(=O)CCc1cccc(C#N)c1 N1(C(CCC2CCN(C(C=CC(=O)OCC)=O)C2)=O)CCC(O)C1(C)C C1(C(=O)NCCCP(C)(C)=O)CC(O)C(O)CC1CNC(C1CC1(Cl)Cl)=O C(=O)(CC(C)(C)C#N)N(CCOCCC(=O)NC(c1ncco1)CC)C c1(OCC)ccc(S(=O)(=O)Nc2cc(Cl)nc3c2c(C)nn3C)cc1C c1(CC(=O)N(C2CCN(C(=O)C=CC3CCOC3)C2)C)cccc2nonc12 N1(C(c2c[nH]c(=N)s2)=O)CC2(CCCC2NC(c2ncoc2C2CC2)=O)C1 C=C=C(C)CC(=O)NCC(C)CN(C(=O)Cc1cccc(CC)c1)C C1(C(C)C)C(C(=O)N(CCO)CCN(C)C)CCN1C(c1ccsc1)=O CCCC(CCNC(c1cc(C2CC2)n[nH]1)=O)C1CC1.C12CCOC(C1)C(=O)N2CC c1(OC)ccccc1S(=O)(=O)N1CCN(Cc2cc(Cl)cc(Cl)c2)CC1CC#N c1(C(N(CCCN(C(=O)CN=S(C)(C)=O)C)C)=O)ccc(C(F)(F)F)c(O)c1 CN1CCC(C(=O)NCCc2cnccn2)(NC(=O)Cn2cnnc2)C1 c1(OC)cc(CN2CC(C)CC2C(=O)Nc2ccc(Br)cc2C)cc2c1OCO2 C1(NC(c2nnnn2CCC2(C)CC2)CCOCC=C)CC2(CCC2)C1 N1(C(C(C)n2cncn2)=O)CC2CCC(NC(c3cccc(F)c3F)=O)CC2C1 CC1C(NC(=O)CCc2ccc(Br)s2)CCN1C(C1CCSC1)=O c1(C(=O)NCC2(C(=O)Nc3cnoc3)CC2)nccc2c1[nH]c1ccccc21 N1(C(C(C)(C)SC)=O)CC2CC2(NC(=O)CC2CCCOCC2)C1 C#CCCCCCC(=O)N1CC(NC(c2cc(N)cc(O)c2)=O)CC(C)(C)C1 c1(C(=O)NC(CNC(CC2ON=C(C)C2)=O)C2CCC2)cc([N+](=O)[O-])cc(C)n1 C1(CCOC)(NC(c2ncn(C)c2C)=O)CCN(C(=O)CC2C=CCC2)C1 N1(C(C(C)OCCOC)=O)CC2(CCN(C(=O)CCCc3ccncc3)CC2)C1 C1(NC(C2C(C(C)(F)F)C2)=O)CC2COCC(C1)C2NC(C1CS(=O)(=O)C1)=O N1(C(C(CCCC)O)=O)CCCC2(CCN(c3ncc4cccnc4n3)C2)C1 N(C(=NCCCCl)NCc1cc(C(N)=O)on1)C1CCC(CC(=O)OC)CC1 Cc1cc(C)c(C(=O)NC(C2(O)CCCCC2)C(=O)NCCc2c[nH]nc2O)o1 c1(C(=O)NC(CCCCNC(CCCOC)=O)C)cn2c(C)cccc2n1 C1(COC)(CO)CCN(C(c2ccc(C)nn2)C(=O)NCC2CCC2)CC1 N1(C(C2C(C)(Br)C2)=O)CCC(CCCNC(=O)Cc2cncnc2O)CC1 N1(C(c2ncn(CC)n2)=O)CCC(C)(C)C(C(=O)NC2CCC2(C)C)C1 c1(-c2cc(-c3n(CC4C(C)C4)nc(C4CCCO4)n3)sn2)c(F)cccc1F N1(C(c2c(CCC)n[nH]c2)=O)C2CCC1C(C(=O)NCCCC(C)(C)C)C2 C(CO)(CO)(CO)NC(C1C(CNC(Cc2cc(C)on2)=O)C1(C)C)=O C1(CNC(Cn2cnc(=N)[nH]2)=O)(CNC(=O)CSC2CC2)CC2CCCC2C1 c1(C(C(=O)N(CC(F)(F)F)CC)C(=O)OC(C)(C)C)cnn(C)c1O C1(c2ncc(CC)s2)NC(=S)N(c2ccc(F)cc2F)C2=C1C(=O)NC(C)C2 C(=O)(C(CC(C)C)C(C)C)NCC1(NC(c2ccc(C3(OC)COC3)cc2)=O)CC1 c1(C(N2C(C(C)NC(=O)CC(=O)NCC3CC3)CCC2)=O)cccc(F)c1O Cc1cc(C#N)ccc1-c1cnc(NCc2ccc(O)c(Cl)c2)c(O)c1 c1(C(N2CCN(C(C34CCC(CC3)O4)=O)CC2CO)=O)csc2ccncc12 C1(CC(=O)NCCN2CCC(NC(c3[nH]c(=N)sc3)=O)CC2)CCCCC1(F)F C1(OCCC)CCCN(C(=O)Nc2cc(C)n(C(C)C)n2)CC1 N1(C(CC)=O)CCCC1C1CCCN1C(=O)C(O)CNC(=O)COCCSC C(=O)(CCC(C)(C)C)NC(C(C)C)C(C)NC(=O)CC1CSCCS1 C(CO)(C(=O)N)NC(C(C1CC1)SC)=O.C12(CC1)CCNC2.N(C)C C1(C(N2CCC(Cc3cc(C)no3)CC2)C(=O)NC)C2CCCCCC12 C(CC(C(=O)N1CCC1CC(=O)N(C)C)NC(=O)C(C)C1CCC1)SC C12(C(N3CC(F)CC(NC(c4cc(CC)no4)=O)C3)=O)CCCCCC1OCC2 c1(CC)ccc(CNC(=O)COC2CN(C(C3(CC)COC3)=O)C2)nc1 N1(C(CC2COCC(C)O2)=O)C2CCC(C2)C1C(=O)Nc1cnn(CCF)c1 C1(CNC(C(CC2CC2)NC(C(C)=CC2CC2)=O)=O)CCC2CC1CO2 c1(NC(CN(C(CC(COC)C)=O)C2CCC2)=O)c(C)cccc1Br C(=O)(C(C)(C)C(F)(F)F)NCC1CN(C(C(Cc2c(OC)cccc2)=O)=O)C1 C1(C2(O)CN(C(C3(C(C)(F)F)CC3)=O)C2)(CNC(C2CCN(CC)C2)=O)CC1 Cn1cc(C(N2CCOCC(NC(c3cnc(N(C)C)nc3)=O)C2)=O)ncc1=O S(=O)(=O)(c1cnc(NCC2CCOC3CC23)c(Cl)c1)N1CCN(S(C)(=O)=O)CC1 C(CCCCN(C(=O)N(C1CCCSC1)CO)C)C(C)C(=O)OC(C)(C)C.C1CO1 Cn1ccc(C(N2CC(C)(OCCC(=O)Nc3nonc3N)C2)=O)c1 c1(C(N2CC(CNC(C(C)=CC)=O)C(O)C2)=O)nccc(Br)c1C Cn1cc(S(=O)(=O)NC2CCN(CC3CC(N)C3)C2)cn1 CC1(C(=O)NC2CC(NC(=O)CC3CC(O)C34CCC4)C2)CC2CCC1O2 c1(C(=O)NC(c2n(CC(C)C)ncc2)(C)C)ccc(Cl)cc1[N+](=O)[O-] c1(C(N2CCC(N(C(=O)CC3CCCSC3)C)CC2)=O)ccc([N+](=O)[O-])c(N)n1 CCCCCS(=O)(=O)CC(=O)NCCCNC(c1nnc(S)n1C)=O C1(N(C(C2(C(N(C(C)C)C)=O)CC2)=O)C)CN(C(=O)C#CC2(C)CC2)CC1(C)C C1(C(N(C)CCNC(=O)CCC2CCOCC2)=O)CCC2(C1)CC2(F)F N1(C(CCSCC(=O)OC)=O)CCCC(NC(=O)CC2CC2(C)C)C1C N(C1CN(C(=O)C=CCCC(C)C)Cc2ccccc21)C(C(C(CC)C)O)=O C1(CNC(C(c2ccsc2)C)=O)CC(C)(C)CN1C(c1cncc2[nH]ccc12)=O C#CCCCC(C)(c1nnnn1CCOCC)NCCn1cc(Br)cn1 c1(C(C(=O)NC2COC2)N(CC#CC)CC)nc(C(F)(F)F)n2c1CCCC2 c1(C(N2CCC(C3CC3)C2CNC(C2(O)CCOC2)=O)=O)nccc2occc12 C1(CNC(c2scnc2C(F)(F)F)=O)CN(C(=O)CC2CCCO2)CC1C(F)F C1(CC(N2CCC(N(C(=O)CN(C)C)CCC)C2)=O)C(=O)NN=C1C c1(C(C(=O)NCc2ncc(C(F)F)cn2)F)ccc(F)cc1Cl C(=O)(CC(C)C(C)(C)C)NCC1(F)CC(NC(c2nc(C(=O)OC)sc2)=O)C1 C1(C(N2CCN(C(C3(C=C)CCOCC3)=O)CC2)=O)CC2(CCCCC2)S1(=O)=O N1(C(COCCCOC)=O)CCC2(C1)CN(C(c1cnn(C3CCOCC3)c1)=O)C2 C1(NC(c2n(CC)ccn2)=O)CCC2(CCCN(C(c3cccnn3)=O)C2)C1 C(C(C)(O)CC(=O)N1CC(NC(c2c[nH]ccc2=O)=O)CCC1C)OC C1(NC(CCCC#C)=O)CCCCCC1NC(=O)C(C)Cc1ccncc1 C12(C(N3CCC4(C(NC(c5ccc(OC)nc5)=O)C4)C3)=O)CCC(N=[N+]=[N-])C1C2 C1(C(c2nnnn2C(C)C)N(c2ccccc2)CC2(COC)CC2)CCCCCC1 CCCC(=O)NCCOCCO.C(C(C)(C)C)=CC(=O)N(CCCO)C C(=O)(CCCCNC12CC(C(=O)NC(C)C)(C1)C2)NC(=O)NC(C(=O)OC)C c1(C(=O)NC2(C(F)F)CC(COC(c3cncc(Cl)c3)=O)C2)cc2c(s1)CCC2 c1(CNC(C(CC)=CC)=O)cnn2c1CN(C(C13CC1COC3(C)C)=O)CC2 c1(N2CCOCC(C)(C)C2)nc(=NCC23CCCC2C3)[nH]c2c1CCCCCC2 C(=O)(CC(O)(C(F)(F)F)C1CC1)NC1C(NC(CCCCCC)=O)COCC1 c1(C(=O)OC)ccc(N2CCN(C(=O)CCC(F)Br)CC2)c(F)c1 CC1CCC(NC(=O)C(C)(C)c2ccsc2)CN1C(=O)C=CCN1CCOCC1 C(=O)(CCCC(C)NC(=O)C(C)CCCC)NC(C#C)CC1CC1 C1(NC(CC2(C)CCOCC2)=O)CC2(NC(=O)C=CC3CCCO3)COC1C2 N1(C(C(C)NC(C)=O)=O)CCN(C2CN(C(c3coc(C(F)F)c3)=O)C2)CC1 Cc1nncn1NC(=O)C12CC1CN(C(c1cc3ccccc3o1)=O)C2 C1(C(N2C(C#C)COCC2)=O)COC2(CCCC2)C1 CCC(CCC(=O)N1CC(C)=CC(C)C1)NC(c1cc(=N)[nH][nH]1)=O Cc1nnc(O)c(C(=O)NC2CC(CNC(=O)Cc3ccc(Cl)s3)C(O)C2)c1C CC1CN2CCC1C2.C12(C(=O)N(C)C)CC(C)(CN1C(C1CC1C(N)=O)=O)C2 C1(NC(c2nc(CCCC)sc2)=O)CC(O)CN(C(=O)C(C)C(C)(C)C)C1 c1(C(=O)NC(C)C(C)(C)NC(C2CCCCN2C)=O)cccc2c1ncn2C CC1Cc2cc(Cl)ccc2N1CC1(C#N)CC2(CC(C(=O)O)C2)C1 c1(OC)ccc2c(c1)CCC2C(=O)NCCCNC(c1cccnc1)=O N1(C(CC(=O)OC)=O)CCCCC1C1(CNC(c2c[nH]nc2F)=O)CC1 c1(C(=O)OCCCC(C)c2cccnc2)ccc2c(c1)CCC(C)(C)O2 N1(C(C(C2CC2)OC)=O)CCN(CC(C)NC(c2cc[nH]c2C(C)C)=O)CC1 O(N(CC)S(=O)(=O)c1ccc(-c2ccncc2)cc1Cl)CC c1(C(=O)NCCCCN(C(=O)C(O)C2CC2)C)c[nH]c2cccc(Br)c12 c1(-c2cccc(C(O)OC)c2)cc(C)cnc1F c1(OC)nccc(C(N2CCC(C(F)C(=O)N(C)CCc3cccs3)C2)=O)n1 CC1CC2(CCN(C(C3CCN(C(C4(C)CCCN4C)=O)C3)=O)C2)CO1 C(CCCN1CCC1)N.CC1CC1CC(=O)NCCCC1(NC=O)CC1 c1(CNC(C2CC(C(C)NC(c3cnoc3C3CC3)=O)C2)=O)ccccc1C#N C=CCCC(C)(C)C(=O)NCC(F)(C(=O)NCCCN1CCOCC1)C(C)C N1(C(c2cc(C(C)O)on2)=O)CCC(O)(C(C)NC(=O)CN2CCOCC2)CC1 c1(C(N(CC(C)NC(=O)C(C)(C)c2ccno2)CC)=O)ccc(O)nn1 N1(C(C2CCC(C(C)C)CC2)=O)CCOC2CN(C(=O)CNC=O)CC12 c1(C(=O)OC)c(F)ccc(NC(C2CC(F)CN(C(c3ccns3)=O)C2)=O)c1F c1(C(N2CC(c3ccccc3)(NC(C(CC=C)C)=O)C2)=O)nn(C)cc1S(N)(=O)=O CC(CC=Cc1ccccc1)C(=O)NC(C)(CNC(=O)CCNC(N)=O)CO C1(C(C)C)(NCc2cc(O)ncn2)CCCN(C(=O)OC(C)(C)C)C1 C1(NC(C(C#C)(C)C)=O)CN(C(=O)COCc2nc(C)no2)CC1N=[N+]=[N-] C1(Cc2ccccc2)CC(C#N)(n2cc(C3(O)CN(C(=O)C4=NOCC4)C3)nn2)C1 c1(OCC)ccc(F)cc1C(=O)NCC1CC1NC(=O)C=Cc1ccc(F)cc1 N1(C(=O)NC(c2onc(CSC)n2)C)CCN(C(=O)C=C(C)C(=O)O)CC1 C1(CC#C)(CNC(c2cc(C(=O)OCC)on2)=O)CC=CCC1 C1(C(N2CCCC(O)(CNC(C3CSC3)=O)C2)=O)(COC)CCCNS1(=O)=O c1(OC)cc(I)c(CN2CC3COCC3(C(=O)NCC#N)C2)cc1OC c1(OC)ccc2[nH]c(C(N3CC4CCCCC4C3C)=O)cc2n1 N1(C(c2onc(C)n2)C)CCN(C(=O)CNCC(O)C2CCC2)CC1 C(=O)(CC(CN(C)C)C(F)F)N(C1CCCN(C(CN(CCC#C)C)=O)C1)C C(=O)(NNc1cccc(Cl)c1C)N1CCC(N(C)C(=O)OC(C)(C)C)C1 Cc1nc(C(N2CCC(CN(C(=O)CC3CC3C(F)(F)F)C)C2)=O)cs1 C#CC1(C(=O)NC2CCCN(C(=O)CCCn3c(O)nnc3O)C2)CCCCC1 c1(C(=O)NC2CCN(C(c3cn[nH]c3)=O)C2)cc(Cl)cnc1Br c1(OCC)cc[nH]c(=NCCNC(=O)C(C)Cc2ccco2)n1 C(=O)(C(O)CC[S+](C)C)N(C(CCNC(CCc1c(C)cccc1)=O)C)C c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)CC2CC)ccnc(N(C)C)c1F C1(CC)(NC(=O)CCc2cncn2C)CCN(C(C2CCC(=O)N2C)=O)CC1 C=CC(C)(CC)C(=O)NCC1(C)CCN(C(=O)C=Cc2ccccc2C)C1 Cc1cc(=O)n(CCC(=O)NC2CC2CNC(=O)C(C)(C)C2CCCC2)cn1 C1(C(=O)NCC2CCN(C(CC3(C)CCC3)=O)CC2(F)F)CCCCC(F)(F)C1 N1(C(c2c(OC)cccc2)=O)CCC2C(CCCN2C(=O)Cn2nccc2C)C1 C1(C(N(C2CCN(C(C3SCCS3)=O)C2)CC#C)=O)CC12CCC2 Cc1[nH]nc(C(=O)NCCC2CCCN2C(c2cccc(N)c2)=O)c1C c12ccc(cc1)NC(=O)N2.c12ccnc(c1)C(=O)N2.c1(C(C)(C)C)cccnc1 c1(COC(c2cc(C)n(-c3ccncc3)c2C)=O)ccccc1[N+](=O)[O-] C12(CNC(c3cc(CC)on3)=O)CCC1CCN2C(c1nc(OC)ccc1Cl)=O C(=O)(NNC(=O)CC(N)c1cccc(Br)c1)c1ccc(C)cc1 c1(OC)ccc(CC(=O)NC2CC(NC(=O)CCNC(=O)CO)C2)cc1.C1CO1 c1(C(=O)NC(C2(O)CN(C(c3ccc(C(F)F)cn3)=O)C2)C)cc[n+]([O-])cc1 Cc1cn2c(CC(=O)NCc3ccccc3OC(C)C)cnc2s1 CC(C)CCC(=O)N(C1CCC(c2cn(CC3CCCOC3)nn2)CC1)C1CC1 c1(C(N2CC(CN(C(=O)CC(F)(F)F)C)OCC2)=O)cccn2nnnc12 N1(C(C(C(C)C)OC)=O)C2CCC1CC(N(C(=O)CSc1ccccc1F)C)C2 C1(CNC(C#CC(=O)N(C)C)=O)CN(C(c2coc(C3CCC3)n2)=O)CCCO1 c1(CN2CC3(C(NC(CC(CC=C)(C)C)=O)CCC3)C2)cc([N+](=O)[O-])ccc1N Cc1cccnc1C=CC(=O)NC(C)CCN(C(=O)Cc1nncn1C)C c1(-c2cn(CCCC(=O)NCCN(CC)CC)nn2)ccc2nc(C)ccc2c1 C1(F)(C(=O)NC2CCC(C)(CNC(c3c(C)nsc3)=O)C2)CCCCCC1 C(=O)(CCC(=O)NCC(C)NC(=O)Cc1sccc1Cl)Nc1nnc(C)s1 c1(C(N2CCCC(CNC(Cn3nnc(C)n3)=O)CC2)=O)ccnc2ccnn12 N1(C(c2c(SC)scc2)=O)CCOC(C(C)NC(=O)CC2CC(C)(C)C2)C1 N1(C(c2cc(Cl)nc(=N)[nH]2)=O)CCCN(C(=O)CN2CCNC(=O)C2)CC1CO C1(CNC(C2C(CC)CCC2)=O)CN(C(c2ccc(C(C)=O)[nH]2)=O)CC(C)(C)O1 C(=O)(C1=Cc2ccccc2C1)NCC(S(C)(=O)=O)CNC(=O)C(O)c1ccco1 C1(C)(NC(C=CC2N(C)CCC2)=O)CCCN(C(C2CCN2C)=O)C1 c1(CNC(C2N(C(CSCC#C)=O)CC2)=O)cncc(OC)n1 c1(C(=O)NC2CN(C(c3c(C)n(C)nc3)=O)C(C)CC2)cccc2ccnn12 CC1CN(C(=O)CC2CCS(=O)(=O)C2)CC1NC(C1(C)CCOCC1)=O Cn1nnc(CNC(C2(C)C=CCC2)=O)c1C(=O)NCC1(C)CC2CC2C1 c1(C(N2CC(NC(=O)C(CO)c3ccccc3)C(F)C2)=O)c(Cl)cc(Cl)cc1Br C=CCC(C)(CC)C(=O)NC1CCN(C(=O)COCc2ncc(C)o2)CC1CO C1(C(N(CCC)CCOC)=O)CC(C)CN(C(=O)C(C)SC(C)C)C1 c1(CNC(=O)NC2C(CC(=O)OC)C2(C)C)cc2c(nc1O)CCCC2=O CCC(C#N)(CC)C(=O)N1CCOC(CNC(C2CC=CCC2)=O)C1 Cc1ncc(C(=O)NC2(C(=O)NCC(c3cn(C)cn3)O)CC(O)C2)cn1 C1(CC=C)(NC(c2scnc2C)=O)CN(C(=O)COC2CC=CC2)C1 c1(SC(C)C(=O)OC)ccc(C#N)cc1.N1(C=O)CC2CC2C1CNC(=O)CC(F)F C(=O)(C(N)CCC(=O)O)Nc1ccc(Sc2ccc(C)cc2)cc1 C=C(Cl)CC(C(=O)N1CC(F)(CC)C1)NC(=O)C(CC1CCC1)OC CC(C)(C)C(CO)C(=O)NC1CN(C(c2ccnn2C2CCC2)=O)CC1N=[N+]=[N-] c1(C(=O)NCCCOCCNC(=O)Cn2ncnn2)cc(F)c(F)cc1F N1(C(C(C=C)(C)O)=O)CCC(C)(CCNC(c2cnncc2O)=O)CC1 C1(NC(CC(C)OC)=O)CCN(C(c2cncn2-c2cnn(C)c2)=O)CC1CO C(=O)(CC(C)(C)CCOC)N1C(C(=O)NCCCCCCC)CCC1 C1(CC)CCCCCN1C(C(=O)NC(C)C)C1CC1 C1(NC(C(C)(C)SC)=O)CN(C(c2cc3ccccc3[nH]2)=O)C2(CCCOC2)C1 N1(C(C2N(CC)CC2)=O)CC(NC(=O)CSc2cccc(Cl)c2)CC(F)C1 C1(C(=O)NCCCCCCNC(C2CC2CF)=O)Cc2ccccc2C1 C1(CC(=O)NC2CCN(OCC)CC2)N(C(=O)CCOC(C)=O)CCC1(C)C N1(C(c2ccc(C3CC3)cc2)=O)CC(NC(C2(F)CCC2)=O)CC12CCCC2 N1(C(C2(F)C(C)C2)=O)CCC(CNC(c2cc(Cl)cn2C)=O)C(F)(F)C1 C(=O)(N1CCC(C(=O)NCC2(F)CC(CO)C2)O1)c1c(C)cncn1 C1(CC)CC(C)CN1C(C1(NC(c2cnn(CC)c2)=O)CCCC1C)=O C1(C(=O)NCC2(NC(c3n(CCC)ncc3)=O)CCC2)CC=CCC1C N12CCN(C3COCC13)C(=O)c1cncc(n1)C2=O.C1(NC)OCCC1C c1(C(=O)NC2CC3(C(NC(C4(C)CC4(Cl)Cl)=O)C3)C2)ccc([N+](=O)[O-])nc1 C(C(C)(C)CC(=O)NC1CC(C(=O)NCC2CC23CCCCC3)C(O)C1)N(C)C Cc1cccc(C(=O)NCCOCC(=O)Nc2ccc(F)c(C(F)F)c2)c1O C#CC1(C(=O)NCC2(O)CC(CO)C2)CN(C(c2ccc(Cl)cn2)=O)C1 N1(C(C2(C)C(C)(C)C2)=O)CCOC(C)(CNC(c2ccnc(OC(F)F)c2)=O)C1 C1(C(CNC(C2(CC)CCC2)=O)(C)O)CCN(C(=O)Cc2csc(CC)n2)CC1 C1(CC)CCCC(NC(C2(NC(=O)CCn3ccnc3C)CSC2)=O)C1 Cc1ccc(CCC(=O)N2CC(CC(=O)NCCCCCl)C2)cc1 C(CCC(=O)NC(C)(C)CN(C)C(C1CCOC1C)=O)=CC(C)C c1(C(c2n(C)nnn2)NCC(C)(C)C)c2ccccc2nn1C c1(CC)cc([N+](=O)[O-])ccc1N1CCC(NC(c2ccnn2C(C)C)=O)C(O)C1 c1(NC(N)=O)cc(NC(N2CCN(c3ccncc3)CC2)=O)ccn1 Cc1csc2ncc(C(=O)NCC3(C)CN(C(c4cscn4)=O)CCO3)c(=O)n12 C1(C(=O)NCC2(NC(c3c(C)c(Cl)ccn3)=O)CC2)CCCN1S(=N)(=O)N(C)C c1(-c2cc(NC(C(n3cc(CCC(C)O)nn3)C)=O)sn2)ccc(F)cc1 C12CCCC1NC(=O)C(F)C1(CC1)C(=O)N(CC)C1(CC1)C(=O)N2.C1CC1.OC C(C1=CCN(C(=O)C(C)(C)n2ccc(C3CC3)n2)CC1)NC(CN1C(C)CC1)=O Cc1cccnc1CC(=O)NC1(C)CCN(C(=O)CCc2ccoc2)C1 CC1(C)CC(NC(=O)C(O)CN2CCCC2)CN1C(c1ncc[nH]c1=O)=O C1(NC(C2N(C)CCOC2)=O)CC=C(C(=O)N2CC(C)(C)C2C2CC2)C1 C(=O)(CS(=O)(=O)Cc1ccccn1)NCCNC(c1n(CC)nc(C(C)C)c1)=O C(=O)(C(CO)C(C)(C)C)N1CC(CCNC(C(C)=CC2CC2)=O)C(C)C1 CC1CCC(C(=O)NCC#CCNC(c2ncoc2C2CC2)=O)S1 C1(C(=O)NCC(C)CN(C)C(c2c[nH]nc2C2CCC2)=O)CCn2cnnc2C1 Cc1cc(-c2noc(CCC(=O)OC(CC(=O)Nc3ccccc3)=O)n2)ccc1F c1(C(=O)NC2CN(C(C(CCC)C)=O)CC2SC)ccc2nc(C(F)F)[nH]c2c1 c1(C(=O)NC2CCN(C(c3cc(C4CC4)on3)=O)CC2)cccn(CCO)c1=O c1(C(N2CC(COC)(NC(C3CCSC3)=O)C2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 C1(NC(COCC(C)C)=O)COC2(CCN(C(=O)CC3CC4CCC3CC4)C2)C1 c1(C(N(C2CN(C(C(C)n3cccn3)=O)C2)C)=O)cncc2nnn(C)c12 Cc1cc(CC(=O)NC2CC3(C2)CN(C(C2CCC2)=O)C3)cc(Br)c1 CC1CN(C(c2c[nH]cc(F)c2=O)=O)CCCN1C(=O)Cn1[nH]cnc1=N CC1C(NC(C2(CCF)CC2)=O)CC2CCC1N2C(=O)C1Cc2ccccc21 CCC(C)(C)CC(=O)NC1CC(C)(NC(c2ncc(N)cc2Cl)=O)C1 C12CCCN(C1)C(=O)CC1CC1CN2C(=O)CSO.c1(C)cccs1.C(CCF)OOC.CS Cc1csc2ncc(C(N3CCC(O)(CNC(=O)CC4CCCC4)C3)=O)n12 c1(SC)cccc(C(=O)NCC)c1.c1(CCC(=O)C2CC2)cnccn1.C1C(CO)N1 C(c1ccc(Br)s1)=CC(=O)OCC(OC)OCCOC N12CCC(C1)NC2=O.c1(NCC(C)N(C)C(C2(C#N)CC2)=O)ccccc1 Cc1ccc(NC(=O)CCC2(C)CN(C(C3(C#N)CC3)=O)C2)cc1C#N c1(-c2nc(C3CNC(=O)OC3)on2)cccc2ccccc12 c1(SC)c(C(=O)NCCOC2CN(C(c3ccc(C)n3C)=O)C2)cnn1C C1(CC)CN(C(C23CC(CC)(CO2)C3)=O)CCN1C(=O)C(c1ccn(C)n1)C c1(N(C2CCC(CO)CC2)C)cc(S(=O)(=O)N2CCCN(C)CC2)ccc1C#N c1(C(N(C)CC2CCCN(C(c3n[nH]c(O)n3)=O)C2)=O)ccc(F)nc1F c1(CCNC(=O)NCC2CC3CCCC3C2)cccc2nccnc12 c1(C(=O)NCCC2N(C(C(=O)NCC(F)(F)F)=O)CCC2)nc2ncccn2n1 c1(NC(C2C(NC(c3cc(Cl)c(Cl)s3)=O)C2)=O)nnc2ccc(Cl)nn12 Cc1c(C(=O)OC(C)(C)C)noc1.C12(OC(c3ccccc3)=O)CC(ON)(C1)C2 c1(C(N(C(CCNC(Cc2nc(C)sc2)=O)C)C)=O)nn(C)nc1C CC1CCN(C(c2ccc(N(C)C)nn2)=O)CC1NC(c1cncn1C)=O C1(CNC(C(C=C)(F)F)=O)CN(C(=O)C=CC2CCC2)C2CCCC2O1 C(=O)(C(C)(O)CC(F)F)N1CCC(CN(C(c2ccc(COC)c(F)c2)=O)C)C1 C1(NC(CCSC)=O)(CNC(c2cnn(-c3ccccc3)n2)=O)CCOC1 CCC(O)C(C)C(=O)NCC(c1ccc(OC)cc1)NC(=O)C=C(C)C(C)C c1(NC(C2CC2C(N2CCS(=O)(=O)CC2)=O)=O)c(Br)cc(Cl)cc1[N+](=O)[O-] C(=O)(CC(C)CC(C)C)NC(C1CCN(C(CCC(C)OCC)=O)C1)C C12(CC(=O)NCC(=C)CCNC(c3ccc(C)s3)=O)CCC(CC1)C2(C)C C1(CNC(C(C)OCC)=O)CC(C(F)(F)F)CCN1C(=O)C(O)CCC N1(C(CCC2CC(NC(c3cc(CCC)on3)=O)C2)=O)CC(C)C(C)C1 c1(OC)cc(OCC(F)(F)F)nn1C.c12ccc(cc1)NC(=O)C1CCC21 C1(CC)CN(C(=O)C(F)n2cccn2)CCN1C(c1cc(-c2ccncc2)[nH]n1)=O C1(C(=O)NCCC2CC(O)C2)C2CCC(C2)N1C(C1(CO)CCCCO1)=O c1(C(=O)NC2(CF)CCN(C(c3ccco3)=O)C2)ccc(F)c(OC(F)(F)F)c1 c1(SCC)c(-c2ccc(-c3nccn3C3CCC(O)CC3)s2)cc(F)cc1F C#Cc1cncc(NC(C2CCN(C)C(=O)C2)=O)c1 N1(C(c2c(C)c(F)cnc2)=O)CCC2CCN(C(c3cncn3C)=O)CC2C1 N1(CC=C)CCCN(C(C2CCCC2CNC(=O)Cn2cnnc2O)=O)CC1 C1(C(N(CC(C)NC(=O)CC=CCc2ccccc2)C)=O)(CO)CC1(F)F C12(NC(C(C)SC)=O)COC(C1)C(NC(=O)Cn1nnnc1-c1ccsc1)C2 c1(-c2ccc(C3C(C(=O)NCc4cnco4)C3)c(F)c2)ccc2c(c1)NCCO2 C12(C(=O)NCCCN(C(C3CC(=C)C3)=O)CCO)COCC1C2(F)F c1(CC(=O)NC2CCN(C(c3cnccn3)=O)CC2F)coc2cc(F)ccc12 c1(C(N2CCC(CNC(C3CCCCO3)=O)C(O)C2)=O)c(F)ccc(F)c1Cl C(=O)(C(CN)C(C)C)NCC(c1cccc(C)c1)O N(C(=NCC1CC=CCC1)NCCN1CCC(OC(C)(C)C)C1)C(C=C)C Cc1ccc(CCCNC(=O)C(N)CCOCC(C)C)cc1 CC(C)C(C(=O)N(C)C)N1CCCCC1C1CCCOC1.C(C)(C)(C)O.C1COC1=O CC(CCOC(F)(F)F)C(=O)NC(c1cnn(C)c1)c1ccccc1 N1(C(CC(C)OC)=O)CCC(NC(=O)CCn2cnccc2=O)CC1C C1(N(C(C(CCC)O)=O)C)CCCN(C(c2cc(C)c(Cl)cn2)=O)CC1 C1(NC(CC2N(C(C3CCCN(CC)C3)=O)CCC2)=O)CNC(=O)C1(C)C c1(CN(C(C2CNCCC2(F)F)=O)Cc2c(C)cccc2)c(Cl)ccnc1Cl C(CCC(C)(C)C(=O)N1CCCN(C(c2cc(C)c(C)o2)=O)C(C)C1)OC C(=O)(CC(C)CCc1ccccc1)NCCC(CNC(C(C=C)(C)C)=O)O CC1C(NC(=O)C2=CC(C)(C)C2)CC2CCC1N2C(=O)CCNC(=O)C=CCl N(C1CN(C(=O)CN2C(=O)CCC2=O)CCc2ccccc21)C(CC(F)=CC)=O c1(C(C(=O)NCc2cccc(Cl)c2)N(C(C(C)OC)C)C)nc(C)c(C)s1 Cc1cc(Cl)ccc1OCC(=O)NCC1CN(C)CCN1C(C1CC1(C)C)=O C1(C(N2CC(C)(NC(C(CCCC)O)=O)C2)=O)CCc2nc(C)cn2C1 CC1(C)CCC(C(=O)NCC2CC2C2CC2)CN1C(C1CCCC1O)=O Cc1c(Br)ccc(C(=O)NC(CNC(=O)C=CCF)C(C)C(C)C)c1N C(C(=O)N1CC(CCNC(C2C=CCC2)=O)C1)(c1cccs1)SC c1(CNC(c2cccc(CN3C(C)COCC3)c2)=O)ccc2c(c1)CCC=C2 C#Cc1ccc(F)c(C(=O)NC2CCN(C(=O)CCC(C)C)C2C)c1 C=CCCC(C(=O)NOCCCC)NC(=O)C=C(C)COC C(C)(CCC(=O)N1CCC(NC(=O)Cn2nnc(-c3ccsc3)n2)C1C)OC C(N=c1[nH]cnc(Cl)c1F)C1(C)CCCCN(C(=O)C2=CCCCC2)C1 N1(C(C(c2cncc(F)c2)C)=O)CCC(CF)(NC(c2cc[nH]c2)=O)C1 c1(CC(=O)OCc2cccc3[nH]ccc23)ccc2cc(Br)ccc2c1 c1(CC(N2C(CNC(CSCC#C)=O)C=CC2)=O)cc(Br)ccc1F c1(C(C2CC2)OC)ccc2c(c1)CCO2.N12CC(C(C(F)(F)F)CC1=O)NC(=O)C2 C1(C(N(CC(C)C)CC(N2CCOCC2CO)=O)=O)CN(C)CCN1C CCC(C)C1(C)c2nnnn2Cc2ccc(cc2)CCN1.C1(SC2CC2)CCC1 N1(C(C(S(CCC)(=O)=O)C)=O)CCc2sccc2C1CNC(C1(OC)CCC1)=O C12(C(=O)NC3CC(CNC(C4CN(C(C)(C)C)C(=O)C4)=O)C3)CCCC(C1)OC2 c1(C(=O)NC2CC(C)N(C(c3cnn(C)c3)=O)C2)cc2c(Br)ccc(F)c2[nH]1 C(=O)(C(CC)C(=O)N1CCC2C(NC(C3CCC3)=O)CC12)OCC CCCC(O)CC(=O)NCC1CCCC(CNC(=O)CNc2ccc(Cl)cc2)C1 C1(N(C(=O)CCS(C)(=O)=O)C)CCN(C(c2cc(N)c(F)cc2F)=O)CC12CC2 C1(NC(c2ccco2)=O)CCC2CN(C(=O)CC3CC4(CC4)C3)CCC2C1 N1(C(C2(Sc3ccccc3)CC2)=O)CCC2CCC(C1)N2c1ncncc1Br c1(CC(=O)OC)sccc1N(C(=O)CCCNCCCNC(C)=O)CC c1(CN2C(CC)CN(c3nc(=N)[nH]c(C)c3Cl)CC2)ccc2c(c1)CCCC2 c1(C(N2CCC(NC(CC(=C)C)=O)C(F)C2)=O)cc2c(C)c(F)ccc2[nH]1 C(=O)(C(CNC(c1cccc(OC)c1)=O)(CC)CC)NCC(CCCC)O C(=O)(CCC(C)(C)C)N(C(C(=O)NCC(CC)(C)O)C1CC1)C c1(CC(=O)OC)ccc(N(C2CC3CNC2C3)C(=O)Cc2cc(C)on2)c(F)c1 N1(C(C(=O)NC2(C)CCNC2)=O)Cc2cccc3c2C(CCC3(C)C)C1 C1(N(C)C(C2CCCN2C(=O)CN2CCCC2=O)=O)CCCC1(F)F C1(C(=O)NC(C2CCCO2)C)CN(C)CCN1C(c1ccon1)=O C(=O)(C(F)(F)C(F)(F)F)N1CCC(CCNC(C(Cc2ncn(C)c2)O)=O)C1 C=CCC(C)(C)C(=O)NCCN(C(=O)C(O)CCC)CCOC C(CCC(=O)NCc1nocc1C(=O)NCc1ncccn1)NC(N)=O c1(CCC(=O)NCC(CNC(c2c(C(C)C)nns2)=O)F)nc2ccccc2[nH]1 C(=O)(C(C)C(O)C(C)C)NCC(CNC(c1c(OC)nsc1)=O)(C)OC C1(OCC)CC2CN(C(=O)C(C3(O)CCC3)NC(=O)CN3C(=O)CNC3=O)CC12 C12(NC(CC3C(CC)C3)=O)CCC(CN(C(=O)C(C)(C)C3CCC3)C1)C2 C1(C)(C(=O)NCC(=O)NCC(=O)N(C)CC2(C)CCC2)CNC(=O)C1 C1(n2cc(C(N(C(c3cn(C4CC4)nn3)C)C)=O)nn2)CCCCC1(F)F CCC(O)C(C)(C)C(=O)NCCCCC(CO)NC(=O)C=Cc1ccco1 CC1CCN(C(=O)C(=O)NC2CN(C(C3CCCC3(C)C)=O)C2)CC1 C1(C)(CNC(C2C(NCC)C2)=O)CCC(NC(c2cc(CC)cnc2O)=O)CC1 CC1CC(C)CN1C(c1cc(CC2CC2)no1)C(=O)NCCC1(C)CC1 Cc1nn(CC(=O)NCC(O)CN(C)C(C2C(Cl)(Cl)C23CC3)=O)c(C)c1C N1(C(C#CC(=O)N(C)C)=O)CC2CC1CC2NC(=O)C=Cc1ccncc1 c1(C(=O)NCC2C=CC(NC(c3[nH]n(C)c(=O)n3)=O)C2)cc2cncn2c(O)n1 N(C)(C1CCc2c(C)cccc21)C(c1ccn(CCF)n1)C(C(CC)(C)C)=O.N c1(CN(CC(C2CCCC(C)C2)CCO)CC)ccc(C)cc1C N1(C(C=CC(=O)NCC)=O)CCCC1CN(C(=O)CNC(=O)CSCC(C)C)C CN1CC(=O)N(CC(N2CCOC(CNC(C3CCCCC3O)=O)C2)=O)C1=O N1(CC)CC(C(=O)N(CCNC(C2(C)CCCCO2)=O)C(C)C)CC1=O c1(C(=O)NC)cc(C)[nH]c(=NCCCNC(C2CNC(=O)N2)=O)n1 c1(C(N2CC(NC(=O)Cc3csnn3)CC(C)C2)=O)cc(F)cc2nc(S)[nH]c12 Cn1c(=O)ccn(CC(N2CCC(NC(c3ccc[nH]3)=O)C(O)C2)=O)c1=O C1(NC2(c3n(CCSC)nnn3)CC3(CC3)C2)CCSC(C)(C)C1 c1(OC)cc(N2CC(O)(CCNC(c3ccnc(F)c3OC)=O)C2)c(C#N)cn1 CC1CCN(CCC(c2ccccc2)=O)C1(C)C C1(NC(c2c(-c3nc(C)sc3)c[nH]c2)=O)CC(CNC(=O)OC(C)(C)C)CC1O c1(C(=O)NCC(C(C)C)(C)NC(=O)CCCCC2CC2)ccc2cnoc2c1 CC(C)C(Cc1ccccc1)C(=O)NC(C)CCN(C)C1CC1 C1(OCCC)CCCN(c2nnc(C3CC3)n2CC2CCCO2)C1 C(=O)(C#CC1CCOCC1)N1C(C(=O)Nc2c(CC)nc(C)cc2)CC1C Cc1cnn(N(CC(O)CF)CC2C(C)CN2C(=O)OC(C)(C)C)c1 C(CC(=O)NCC1=CCCC1)(C1CC1)NC(c1cc[nH]c1)=O c1(CC)cc(C(N2CC(CN(C)C(c3csc(C)c3)=O)C3(CC3)C2)=O)c(C)nn1 c1(C(N2CC(NC(C(C)OC3CCCC3)=O)C(CO)C2)=O)cccc2ccsc12 C1(CNC(C(CCCC)C)=O)CN(C(=O)C(C)N(C)C)CCC1(C)C N1(C(C=CC(=O)OCCCC)=O)CCC(C)(CNC(c2c[nH]c(C(N)=O)c2)=O)C1 C#CCC(CC(F)F)C(=O)NC(C)CCCCNC(c1cc(OC)cnc1F)=O c1(C(=O)NCC(CNC(c2cc(OC)no2)=O)(C)O)c(C)[nH]c2ccccc12 c1(C(=O)NC2CC3N(C(CSCCC)=O)C(CC3)C2)ccc(=O)n2c1CCC2 c1ncc(Br)c(O)n1.c1(C(N(C2CCN(CC)CC2)CC)=O)c(C(F)F)cnn1C C#CCC(CC#C)C(=O)NC1CCC(NC(C2CC(CC)=NO2)=O)CC1 C1(CNC(C(CCSC)O)=O)CN(C(=O)COc2ccc(F)cn2)C(C)(C)C1 C1(O)(CNC(c2c(C(=O)OC)coc2)=O)CCCN(C(=O)CCCCCF)C1 C1(N(C)C)CC2CC1CN2c1nc(C(=O)O)c(Cl)s1 C1(C(=O)NCCCN(C)C)(NC(Cc2ccc(C)nc2)=O)CCC(C)(C)C1 C12(CC(=O)NCC3CC(CC)C3)CCC1CN(C(=O)CN1CCCCC1)C2 c1(C(=O)NCC2(OC)CN(C(=O)CS(N)(=O)=O)C2)cc(F)c(F)c(F)c1F C(C1C(=O)N1C)N(C)C.C1(C(=O)NC2(C(=O)N(C)C)CC2)CCC1C(N)=O Cc1nc(C)n(CC(=O)N(C2CN(C(C3CCC3c3nc(S)n[nH]3)=O)C2)C)n1 C1(NC(C)=O)CCC(C)(CNC(=O)CCC(=O)N2CCOCC2)C1 CC(C)(CS(C)(=O)=O)C(=O)N1CC(NC(C2CC23CC(F)(F)C3)=O)CC2(CC2)C1 C(=O)(CC1=CCCC1)NCC(C(C)C)NC(c1c(C)sc(O)n1)=O Cc1c(C(N2CCC(C)(CNC(C3CSCCS3)=O)C2)=O)oc2ccccc12 C1(NC(c2cc(OC)c(O)nc2)=O)CC2CC1CN(C(=O)C(C)CC1CCC1)C2 C1(NC(COCCCOCC)=O)CC(C)CN(C(=O)C(CC)CC)C1 c1(-c2ccc(OC)nc2)n[nH]c2ccc(C(=O)NC(c3cccc(F)c3)C)cc12 c1(C(N2CC3C(C(N4CCC(OCC)CC4)=O)(C3)C2)=O)cc(C)n2ccnc2n1 c1(C(N2CCOCC(F)(CNC(C(C)=C(C)C)=O)C2)=O)cccn2c(C)nnc12 c1(C(N2CCC(NC(CC3(C)CCCCC3)=O)C2(C)C)=O)nsc2ccccc12 O=C(C(O)CC1CCCCC1)NCC(F)CNC(c1nncs1)=O c1(CN(C)C(C2CCC3(C2)N=N3)=O)cccc(CNC(C2CCN2C)=O)c1 N1(C=O)CCC(C(=O)NC2(CCC)CCC2)C(C)(C)C1.C12(CCC1)C(=O)O2.[SH](=O)CC Cc1ccc(Br)c(C(N2CCOCC2CNC(c2cc(Br)cnc2F)=O)=O)c1F c1(NC(C(=O)NCc2ccc(CC)cc2)=O)cc(C)nc(C#N)c1 N1(CC(CC)O)CC(C(=O)OC)(Cc2cnn(CC3CCCC3)c2)C1 c1(NC(c2nccs2)CC)nc(=NCC2CCOC(C)(C)C2)[nH]c2ncn(CC)c12 N1(c2cncc(Cl)c2)CCCC12CCOC2 c1(C(=O)NC(C(C)C)CCN(C)C(c2ccns2)=O)ccc(F)c(S(C)(=O)=O)c1 Nc1cncc(-c2cn(Cc3cccc(CNC(N)=O)c3)nn2)c1 c1(OC)cc(C)c(CN2CCOC(C(C)C)(CN(C)C)C2)cc1OC c1(C(=O)NCC(C(C)C)NC(=O)CC2CCCCO2)cncc([N+](=O)[O-])c1 c1(OC)ncc(C(N2CCC(CC(=O)N(C3CCC3)C3CCC3)CC2)=O)cn1 C1(C)(C(C(=O)CN)=O)CCC(=O)C1.CCCC(C)CNC(=O)CN C1(CNC(C(CN(CC)CC)F)=O)C2CCCC1N(C(=O)CC1CN(C(C)=O)C1)C2 C1(C(=O)NCCC2(NC(COCCOC)=O)CC2)CCC(NS(=O)(=O)C(F)F)C1 C#CCCN=c1scc(-c2ccc(C)cc2)n1CC1CC(OC(F)F)C1(C)C CC(C)C(CC(=O)N1CC(C)C(F)C1)NC(=O)CC1CC(=O)NC1=O c1(NC2OCCN(S(CC)(=O)=O)CC2)ccc(N2CCCC(C)C2)c(F)c1 C1(CNC(C(C)N(C)C)=O)CCC12CCN(C(=O)Cn1cnc([N+](=O)[O-])n1)CC2 Cc1noc(C)c1CC(=O)NC1CN(c2cc(-c3ccccc3)ncn2)CC1F C(C(C)NC(c1cccnc1OC(F)F)=O)(C(C)C)NC(C=CCCC)=O c1(C)ccc2c(c1)OCO2.Cc1cnn(CCO)c1C(=O)OC1CC1C C1(CNC(=O)C(=Cc2cn[nH]c2)C2CC2)CN(C(C23CCN(CC2)C3)=O)CCO1 Cc1nc2nc(=S)[nH]n2c(C)c1CCC(=O)NC1CC1NC(=O)C(F)CC1CC1 C1(C(=O)NCCC2CCCN2Cc2sncc2Br)C(C(F)(F)F)C1[N+](=O)[O-] c1(C(=O)NCC2CC(C)N(C(=O)C(C)N(C)C)C2)cc2nn[nH]c2cc1F C(=O)(CCCCCCC(=O)NC1(O)CCN(C(=O)C2=CC=NC(=O)C2)C1)OC C1(NC(c2cccc(C)c2)=O)CCN(C(=O)CC(C)N(C)C)CC1C CC(C)C(C(=O)NCC(C)(O)CNC(=O)CO)N1CCCCC1=O C(=O)(C1COc2ccccc21)N1CCC(N(C(c2c(OC)cc(F)cc2)=O)C)C1 C1(CC)CCCC(NC(c2cc(CNC(C3CCC4CC34)=O)nn2C)=O)C1 C(C1CN(C(c2cc[nH]c2)=O)CC1C(=O)NCc1cccc(CO)c1)=CC C1(COC)C(=O)NCCN1Cc1cccc(-c2cccnc2)c1 CCC(CC)C(=O)N(CCCCNC(=O)C(c1cnn(-c2ccccc2)c1)=O)C C1(C(N)=O)CC(F)(F)CN1C(c1cc(-c2cnoc2)cnc1F)=O Cc1n[nH]c(C)c1CC1CCCN(C(c2ccc(Cc3ccccc3)[nH]2)=O)C1 O=C(C1=CCCN(C(=O)CC2CC2)C1)NCCCc1ccc(Br)cc1 N1(C(COC)=O)CCC(c2cn(Cc3ccc(Br)s3)nn2)C12CC2 C(=O)(C(CC(C)C)NC(C1CCC12CNC2)=O)NC(C(=O)OC)C CN1CC=CCC1CC(=O)NCC(c1ccccc1)NC(=O)Cc1ccn(C)n1 c1(C(=O)NC2CCC(NC(CC3(OC)CCC3)=O)C2)cc2c([nH]1)CCC(C)C2 NC(=O)CC(O)C(=O)NCC1(CNC(=O)CCCC(=O)NC2CC2)CC12CCC2 CC(CCCNC(=O)C(C)SC(F)(F)F)NC(C1CCCSC1)=O C1CCCCCC(c2nnnn2C(C)CC)N1.c1(COC)nc(C(N)=O)no1 C1(NC(=O)C=CCn2cncn2)CN(C(c2ccc(F)cn2)=O)C2CC12 N1(C(C(c2ccccc2)N(C)CC2CC2)=O)CCCC1(C)c1ccccc1 c1(C(N2CCC(C)(NC(CN3C(C)CCC3)=O)CC2)=O)cc(F)cc2nc(S)[nH]c12 CCC(CC(C)C)C(=O)NC1CC(F)CN(C(c2cnc(-c3ccco3)s2)=O)C1 C1(C(=O)NCCCN(C(C(C)SC)=O)C)C2CCC1(C)C2(C)C C(=O)(C1=C(C)CCOC1)N1CC(C=C)(CC(=O)NC2CCN(C(=O)CC)CC2)C1 n1(CC)ncc(C(=O)NCC(N2CCCCC2CF)=O)c1C CCC(CC)CC(F)C(=O)N1CCCC1C(=O)NC1CCOCC1 CC(C)CC(C)(O)C(=O)NCC1CC(C(N2CCC(O)(C(F)F)C2)=O)C1 N1(C(CC2(C=C)CCC2)=O)CCc2c(CNC(c3cscc3F)=O)cccc2C1 C1(CC)CCN(C(c2cnc(O)o2)=O)C(C(=O)NCC=CBr)C1 N12CCOCC(C1)C(=O)OCC(=O)N(CC)CC2=O.C1(COC)CCC1 c1(C(C)OC(=O)Cc2cnn(CCN(C)C3CC3)c2)cccc(OC(F)F)c1 c1(C(N(C(C)C(C)C)CC(C)C)=O)ccc(NCC2C3CN(CC(C)C)CC23)cc1 N1(C(C2ON=C(C)C2)=O)CCC(C)(CNC(c2ccc(C)nc2N)=O)CC1 Cc1c(C(=O)NCC(C2CC2)N(C(=O)CC2OCCCC2(C)C)C)cncc1N CCCCC(C)C(=O)N1CCCC(CN(C(=O)CN(CC(C)C)CC)CC)C1 C1(CC)(NC(C2CN(C)CCO2)=O)CCN(C(c2cn(C3CC3)nn2)=O)CC1 N1(C(C)=O)CC(N=c2[nH]c3c(c(=NCC(C)CC(C)O)[nH]2)SCC3)C1 C(C)(CN=c1cc(C)nc(OC)[nH]1)NC(CCCC#CC)=O N1(C(c2ccn(C)n2)=O)CC2CN(C(c3ncn(C(C)(C)C)n3)=O)CC2(C)C1 C1(NC(C(C2CCN(C)CC2)N)=O)CCCN(Cc2ccccc2)C1=O C1(CNC(Cc2ccc(CC)c(F)c2)=O)COC(C)(C)CN1C(c1cnn[nH]1)=O C#CC1(C(N2CCCCCC2)=O)CCN(C(c2cc(OC)n[nH]2)=O)C1 c1(CN2CCCC(O)(CNC(C(CC)C)=O)C2)ccc(O)c(C)c1O C1(NC(C(OC)OC)=O)CN(C(c2c[nH]nc2Cl)=O)C2CCCC12 c1(C(N2CC(O)(CNC(C(C)OCCOCC)=O)C2)=O)cc(F)cc2ccoc12 C(c1ccccc1Cl)=CC(N1C(CN(C(c2cc(CO)on2)=O)CC)CCC1)=O N1(C(C2(NC(C)=O)CC2)=O)CC2CC1CN2c1nnc(NS(C)(=O)=O)s1 C(c1cncnc1O)=CC(=O)NCC1(F)CCN(C(C2N=C(C)SC2)=O)C1 C1(C)(C(=O)OCCCNC(CN(CCCOCC)C)=O)CC=C(C)CC1 n1(CC)nc(C(=O)NCc2cc(C(N3CC(O)(C(=O)OC)C3)=O)on2)cc1O CCC(C)(C(=O)N1CCC12CN(C(=O)Cc1ccc(O)cc1)C2)C(N)=O C1(C(=O)NC(C(=O)NC(CCC=C(C)C)C)c2cccs2)CCOC(=O)CC1 N1(C(C(C)OC)=O)CC2CC(NC(=O)C=CCN3CCC3)C(C2)C1 c1(C(=O)NCCC(C)NC(COCC(=C)C)=O)ccc2c(c1O)CCCC2 Cc1cc([N+](=O)[O-])cc(Br)c1OC1CCN(C(=O)CCC(CF)CF)C1 C(N=c1[nH]cc(Cl)c2nccnc12)c1c(C#N)ccc(Br)c1Cl CCCC(C)(CC)C(=O)NC1CN(C(=O)CC2CCC(C#N)C2)C1 N1(C(=O)C=Cc2ccc(Cl)cc2)CCCC2(C1)CN(C(C1CCCC1(F)F)=O)C2 C1(CNC(c2nc(N(C)C)oc2)=O)CC(C)CN(C(=O)CCC2CCN(C)C2)C1 C=CCCCCC(=O)N1CCC(N(C(=O)C(CCOC)OC)CCO)CC1 C1(C(=O)NC2(CNC(COCC(=C)C)=O)CCCC2)CCC2(CCC2)CC1 C1(NC(CC2CC(C)OC2C)=O)CCN(C(C2CC(=O)N2)=O)CC1C C(CCC(CO)NC(C1(O)CCC1)=O)NC(CCc1n(C)cnn1)=O N1(c2nccc(OCCC)n2)CCC(C)C(NC(=O)C(C2CCCC2)OC)C1C c1(Sc2c(C(=O)OC)snn2)nc(C)c(C)[nH]1 c1(CN2C(C(=O)Nc3cccnc3Cl)CNCC2)c[nH]c2c([N+](=O)[O-])cccc12 c1(OC)cc(C(=O)N(C2CN(C(=O)C(C3(O)CCCCC3)OC)C2)C)n(C)n1 Cc1cc(C(N2CC(O)CCC2C(=O)NC(C)CF)=O)cc(Br)c1 C(CC(C(C)(C)C)NC(=O)Cc1nccn1C)N(C)C(c1cc(Cl)ccc1N)=O C1(C)(CNC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)CCc2cc(Cl)no2)CC1 c1(OC)c[nH]c(C(=O)NCC2CC2NC(c2cc(C)n(C)n2)=O)cc1=O Cc1nc(C(N2CCC(C)(NC(=O)COC3CC(F)(F)C3)C2)=O)[nH]c1C C1(CN(C(Cc2cc(CC)no2)=O)C)CN(C(=O)CC(CC)OC)CCO1 C(=O)(C(C)(C)C(F)(F)F)N1CCCC(Cn2cc(C(CC)N(C)C)nn2)C1 CC1(C(N2CCC(NC(C3(F)CC=CC3)=O)C(CO)C2)=O)CCCCCCC1 c1(OC)ccccc1CN1CCC(CNC(=O)CNC(C)=O)C1 CCCCC(C)C(=O)NC1CC12CC(NC(c1cncc(C(F)(F)F)n1)=O)C2 Cc1ccc(CC(C)NC(=O)N(C)C)c(C)c1.c12ncc(s1)CC(=O)N2 CCC(CC(F)F)C(=O)N(CCNC(c1ccnnc1C)=O)C1CC1 N1(C(C2C(C)C2C)=O)CCC2(CN2)c2ccccc21 O=[N+]([O-])c1cc(Br)c(F)cc1NCCN1CCCC(OC2CCOCC2)C1 c1(NC(C2C(C(=O)NCC(F)(F)F)C2)=O)cnc2ccc(Br)cc2c1 N1(C(C2CC(C#C)(O)C2)=O)CCN(C(c2ccnc(COC)c2)=O)C(C)C1C c1(SCC=C)ccccc1C(=O)NCC1(C)CC(NC(=O)CCC2CC2C)C1 C1(N(C(c2cc(CC)no2)=O)C)CC2CC1N(C(=O)Cc1cccc(OC)c1)C2 c1(N(C(c2cnccn2)=O)C2CC2)ccc(CCc2ccccc2)cc1.O=C1CO1 c1(C(=O)NC2CN(C(C(CC)C#N)=O)CC(C)C2)c[nH]c2c(Cl)cccc12 C1(C(=O)NCc2scc(CNC(CN3CC(C)(C)C3)=O)n2)OCCC1(C)C c1(C(=O)NC(CNC(C(C)N(C(C)=O)C)=O)C(C)(C)C)ccc2nnn(C)c2n1 c1(C(N2CC(NC(CC(C=C)C)=O)C(C)(C)C2)=O)cc2sc(C)cc2o1 C(=O)(C1CCCc2cccnc21)NC1CC2CN(C(COCC#C)=O)C(C1)C2 c1(N(CCOC)CCNC(=O)C(C2CC2)OC)nc(C)cc(C#N)n1 c1(C2NC(=O)N(c3c(C#N)cc(F)cc3)C2=O)ccc2c(c1)CCC2=O c1(C(NOCCC)=O)coc(C(C)NC(C2(C)CC(C)C2)=O)n1 CCCCC(O)C(=O)c1ncc(Br)c(C(F)(F)F)n1.C12CN(C1)C2 C(CC(C)(C)C)(C(=O)NCC(c1ccc(C)cc1)NC(C1CSCCS1)=O)OC c1(C(N2C(C)CCN(C(CCCC)=O)CC2)=O)ccc2c(c1)C(=O)NC2 CC1CCOCC1C(N1CSCC1C(=O)NCCC1CC(=O)N(C)C1)=O N1(C(c2c(C)cncc2)=O)CCC2CN(C(c3cnc(S)[nH]3)=O)CCC2C1 S(=O)(=O)(C1CCCCC1)NC1C2CN(C(=O)CCc3cc(F)cc(F)c3)CC21 N1(C(c2cc(COC)no2)=O)CC2CC1CN(C(c1cncc(C)n1)=O)C2 CN1CCN(C(=O)CN2CCSCC2)CC1C(=O)NC1CCC1(C)C Cc1ccccc1SCC(N1CCCC1(C)CNC(C1CCCCN1C)=O)=O CC(F)(F)C(C)(C)C(=O)NC1CCOC1C(N1CCCC(O)CC1)=O S(=O)(=O)(c1ccc(NC2CCSC(C)C2)nc1)NC1C(OC)CCC1 CC(C)C(F)(CNC(C1(NC(N)=O)CC1)=O)C(=O)N1CCC(F)(CF)C1 N1(Cc2c(C)c(O)ccc2)CCc2[nH]nc(C(=O)Nc3cccc(I)c3)c2C1 C1(CNC(=O)Nc2cnn(-c3ccccc3)c2C2CC2)CCCC12CCC2 C1(NC(=O)C(F)Cl)CCCCC12CN(C(C1CCCCO1)=O)CCO2 C1(CNC(C2C(C)C2)=O)CC2(CCN(C(=O)C(=Cc3cccnc3)F)CC2)C1 CC(C)C(O)CCNC(=O)C(CO)NC(=O)C(C)(C)CNC(N)=O Cc1ccc(F)c(C(=O)NCC(C)(C)CN(C(=O)C(CO)N(C)C)C)c1F c1(NC(C2C(O)CCN2C(c2ccc(O)cn2)=O)=O)cc([N+](=O)[O-])ccn1 c1(OC)cc(OC)cc(NC(C2CCCN(C(c3c(F)cncc3F)=O)C2)=O)c1 c1(OCC)nccc(C(N2CC=CC2CNC(=O)CC2(OC)CC2)=O)c1F N1(C(c2c(C)ccc(O)c2)=O)CC2(CCN(C(=O)CCC3CCCN(C)C3)C2)C1 Cn1nc2c(c1C(N1CCOC(O)C1)=O)CN(C(c1cccc(Br)c1F)=O)CC2 C1(OC)CCCC1C(N1CC(C)C1C(=O)N(C)CC1(F)CCCC1)=O N1(CCC)CCC2(CC1)CC2NC(=O)CCC(C)(F)F C1(C(=O)NCCC(=O)N(CC)CC)CC=CC(NC(c2c[nH]c(=N)o2)=O)C1 C1(CC)CCN(C(c2ccc(C#N)[nH]2)=O)C(C(N2CC3CCC2CC3)=O)C1 c1(COCC)nc(C(=O)NCC2CCN2CC(C2CC3(CC3)C2)=O)cs1 N1(C(C(=O)N(CC(C)N(C(C(CSC)OC)=O)C)C)C)CCCCCC1 c1(C(=O)NCC(CC)NC(=O)C=C=C(C)C)ncccc1OC(F)F C(CCCC(=O)NC1CCN2CC12)N(C)C(c1nnsc1N)=O N1(C(C(c2ccco2)NC(c2cccnc2)=O)=O)CCCC1C1CC1 c1(C(=O)NC2CCC(NC(C(C(C=C)C)C)=O)CC2)c(C)ccc2nsnc12 C1(C(=O)NCCC(CCNC(CS(CC)=O)=O)C)(OC)CCC(C)(C)CC1 C1(C(=O)NCCC(=O)OC)CCN(C(c2ncncc2N)=O)C1C(C)C C(C(C)(C)S(C)(=O)=O)c1nnc(N(CCOCC)CC)n1Cc1ccccn1 O(N=Cc1ccc(OC)cc1)CC.C1=CC(=O)Nc2cccc1c2 c1(-c2nnc(N3C4C(C)(C4)OCC3)n2CC(=O)NC2CC2)n[nH]c2c1COCC2 N1(C(C2C(=C)C2)=O)CCC2CC2(C(=O)Nc2cc(CC)cc(F)c2)CC1 N1(C(C(C(=C)Cl)(C)C)=O)CCC2(CCC(NC(c3ccn(C(C)C)n3)=O)CC2)C1 C1(NC(CC=CCNC(CN(C)C)=O)=O)CCCC1(C)O N1(C(CC2OCCN(C(C(C)OCCC(C)C)=O)C2)=O)CCC2(CCO2)C1 C(C(N=[N+]=[N-])C(=O)N1C(CC(=O)NCCCOCCO)C2CCCC12)OCC C1(C(=O)NCCCC(C)NC(CN2CCC(C)CC2)=O)CCC(C)(C)CO1 CCCCCCCC(C(=O)NC(c1ccccc1)C)N1CCC2CCCCC12 CC(C)CC(C)(C)C(=O)NC1CCC1NC(c1ccn(-c2cnccn2)n1)=O c1(C(=O)NCC(CNC(C(C2CCOCC2)OC)=O)O)cc2nc(C)ccc2o1 Cc1nc(C(N2CCC(N(C(=O)Cn3nccc3C)C)C2)=O)c(C)s1 C1(NC(CSCC=C)=O)CCCC(NC(c2nc(-c3cccs3)oc2C)=O)C1 N1(C(c2ccc(C)c(C)c2O)=O)CC2CCCC(NC(c3ccco3)=O)C2C1 CC(C)CCC(O)C(=O)N(C1CCN(C(=O)C(F)(F)C2(O)CCC2)CC1)CCO N1(C(C(C(C)C)N(CC)CC)=O)CCCN(C(C2COCC(C)(C)O2)=O)CC1 N1(C(CCSCC)=O)CCC(C)(C)C1C(N1CCCC(CCC)C1)=O C#CCC(CC(F)F)C(=O)N(CC(=O)NCc1ncn(CC)n1)C(C)C c1(C(=O)NCCCN(C)C(C2NC(=O)CC2C(F)(F)F)=O)cn(C)nc1O c1(C(=O)NC2C(COC)C2)n[nH]c2cc(C)ccc12.N12CC(C(C(F)F)C1)C2=O C1(NC(c2c(C)noc2)=O)(CO)CCN(C(c2ncoc2C2CCCO2)=O)CC1 C1(NC(c2ncccc2Cl)=O)CC2CN(C(C3CCS(=O)CC3)=O)CC2C1 C(C(O)(C1CC1)C1CC1)NC(C=CCC(=O)NC(C1(C2CC2)CC1)C)=O.CSC c1(C(=O)NCC(CN(C(C2C(OC)C2)=O)C)(C)C)ccc(NC(C)=O)cc1O c1(CC(=O)NCC2C(NC(c3cc(CCC)ncc3)=O)C2)c(C)ncnc1C C1(C)(CNC(CCOC)=O)CCN(C(=O)CSCc2ccccn2)C1 N1(C(c2n(CC)cnn2)=O)CCOCC(CNC(c2ccc(Cl)cc2)=O)C1 C1(CNC(C2C(COC)C2)=O)(CO)CCN(C(=O)C(C)(C)c2nncn2C)C1 C1(NC(=O)CCc2cnc[nH]2)CC2CC1N(C(c1cn(C(F)F)cn1)=O)C2 C1(O)(CNC(CN2CCC(C)(O)C2)=O)CCN(C(=O)C=CC=C(Cl)Cl)CC1 c1(C(N2CCC(O)(CCNC(=O)C3=COCCC3)C2)=O)ccc2c(c1)CCCO2 C(=O)(CC(CC1CC1)NC(=O)CC1CC1C1CC1)N(C(C(=O)OC)C)C1CC1 C(=O)(C(C)(C)CCC)N1CCC(C(C)NC(C2C(CCOC)C2)=O)CC1 CCC(C)(C(=O)N(CCCCCNC(C1CC(CCO)C1)=O)C)C(N)=O N1(C(c2nc(C)oc2)=O)CC(NC(c2cc(O)nn2C)=O)C2CCCC12 CN1CCC(C)(CC(=O)NC2(c3nc(NC(=O)CS(C)(=O)=O)no3)CC2(C)C)C1 S(=O)(=O)(CC(=O)N1CCCC1C1CCN(C(C2CC(C(=O)OC)C2)=O)C1)NC c1(C(N2CCC3(NC(CN(CCC)C)=O)C(CC2)C3)=O)cc(O)cc([N+](=O)[O-])c1 CCCCCCCC(=O)N1CC2CN(C(=O)COc3cnn(C)c3)C2C1 Cc1nnc2n1C(C(=O)N(C)CCNC(=O)CSC)CC2.c1(C(=O)N)ccc(Cl)cc1 c1(CC(=O)OC)ccc(NCC(C2CC2)NC(c2cnsc2)=O)c([N+](=O)[O-])c1 C1(C(=O)NCCC2CCN(C(c3n(CC)ccn3)=O)C2)CC2OC(C)(C)OC2C1 O(N1CCC(C(=O)NCC2(CNC(C3CCCO3)=O)CC2)CC1)CC CC1CC(N(C)C(c2n[nH]cc2CNC(C2CCCC2C2CC2)=O)=O)CC(C)O1 C(=O)(C1CCCc2ccccc21)NC1(C2N(C(CS(N)(=O)=O)=O)CCC2)CC1 C1(CNC(C(CCC)N(C)C)=O)CCC2(CN(C(C3COC4COCC34)=O)C2)O1 C1(SC)CCn2cc(CNC(=O)C(C)=C3CCC3)nc2C1 C1(OC)CC(CNC(=O)CCSC)N(C(=O)CCCOc2ccc(C)cc2)C1 C(=O)(N=c1ccn(Cc2cc3ccccc3s2)[nH]1)N(CC)CC c1(C(=O)NC(C(=O)N(CC#C)CC2CC2)CC2CC2)c(C)[nH]c(C)c1C c1(C(=O)NC2(C3N(C(CC4CC(SC)C4)=O)CCCC3)CC2)cncc(Cl)c1Cl c1(C(=O)ONCCC2CCN(CCC=CC)C2)ccc(F)c(C2CC2)c1 C=C(C)CCC(=O)NC1COCCC1NC(=O)C(O)C1CCCC1 c1(CC(N2CC(F)(C(C)NC(C3CCOCC3(C)C)=O)C2)=O)ccc(C#N)cc1F Cc1ccc(C(=O)NCC23CC2CN(C(=O)CCC2CCCOC2)C3)c(F)c1Cl C1(C(=O)NC(c2nnc(O)o2)C)C2CCCC2CN1C(C1CCOC1(C)C)=O N1(C(C2(COC)CCCO2)=O)CC(NC(=O)CSC2CCOCC2)CC(F)C1 N#Cc1cnc2c(F)cc(F)cc2c1NCC1CCC(N2CCOCC2)CC1 C1(CNC(c2cn(C)nn2)=O)CN(C(=O)C(C)(C)C2CCCO2)CCC1(F)F c1(OC)cc(O)ncc1C(N1CC2CCC1(CNC(=O)C(C)(F)F)C2)=O C1(C(=O)NCC(C2CC2)NC(c2ncccc2C(F)F)=O)CCC2CC1CO2 N1(C(=O)NCCC)CCCC1C(=O)O.N1(CC)CCCCC1=O S(=O)(=O)(c1cccc2cccnc12)NC1CCCCN(C(COC(C)(C)C)=O)C1 C1(NC(C2(C(C)NC(C=CC=CC)=O)CC2)=O)CCC(F)(F)C1 C1(C(=O)NC(c2cncnc2)C)CCN(C(c2ccncc2F)=O)CC1O C1(NC(=O)Cn2nnc3c2CCCC3)CN(C(C2COC2)=O)C2(CCCC2)C1 N1(CC(=O)N(C2CCN(C(=O)C(=O)NCC(F)F)CC2)CCC)CCC(C)(O)C1 C1(NC(C2(N(C(=O)Cc3cnc(C4CC4)[nH]3)C)CC2)=O)C2CCCC1CC2 c1(C(=O)NC2CC(=O)NC2)cnc2c(c1)CCN(Cc1ccc(Br)cn1)C2 N1(C(c2ccc(C)nn2)=O)CCCC2C1CCN2C(c1cc(C)c(C)o1)=O CN(C)S(=O)(=O)NCC(=O)NC1(CO)CN(C(c2ncc[nH]c2=O)=O)C1 S(=O)(=O)(c1ccc(NCCCNC)c(Cl)c1)NC(c1cnc(CC)s1)=O C1(CNC(CNS(NC)(=O)=O)=O)CN(C(c2cc(N)ccn2)=O)CC(C)(C)C1 c1(OC)cccc(C(F)C(=O)NCCC(C)NC(=O)C(C)Sc2ccccc2)c1 C1(C(N(CCCOCCNC(C(CC)c2cccnc2)=O)C)=O)CC2CCC1O2 C1(C(=O)NCc2nn(C)c(C(=O)NCC34CC(F)(C3)C4)c2)Cc2ccccc2C1 C1(C(N2CCC(C(=O)NCCc3cn(C)cn3)(CC)C2)=O)CCCC(=O)CC1 CCC(CC(=O)N1CCOCC1CCO)NC(=O)Cc1cnn(C)c1C c1(C(N2CC(NC(COCCCC)=O)CC3(C2)CC3)=O)nc2ccccc2[nH]1 c1(CCC)cccnc1C(=O)NCC1(CNC(c2ccccc2OC)=O)CCC1 C(C(=O)N1CC(O)CO1)(C1CC1)NC(c1cnc(CO)nc1)=O Cc1c(C(=O)NCC2CCCC2NC(c2ccc(Cl)cn2)=O)oc2ccccc12 c1(C(=O)N(C2CCC2(C(=O)O)C(=O)O)CCC(N)=O)cc(C(F)(F)F)co1 CC(C(C)(C)C)N(C)C(c1c[nH]nc1CCNC(=O)CCc1cnco1)=O C1(C(N(CCN(C(c2n(CC)ncc2C)=O)C(C)C)C)=O)CCC2CC1CO2 N1(C(N(C)C)=O)CCC(C(=O)NCCCN(C(=O)C(O)C2CC2)C)CC1 c1(CNC(COC)(C)C)ccc(-n2nc(C)cc2C)nc1 C1(C(=O)Nc2c(OC)nc(-c3ccccc3)cc2)CN(c2nnco2)CC(F)(F)C1 c1(-c2ccco2)cccc(NC(C2N(C(CNC(=O)CN3CC4CC34)=O)CC2)=O)c1 C#CCCC(O)C(=O)NC1(C2CN(C(=O)CNC(=O)CCCCO)C2)CC1 O=C(C#CC1CCOCC1)NC1C2CC1N(C(=O)CCc1cnc(C3CC3)o1)C2 n1(CCOCC)nc(-c2nc[nH]n2)nc1C1(OCC)CCCCC1 C=C(Cl)CCC(=O)NC(C1CCCCN1C(=O)COCC)C N1(C(C2CN(C)C2)=O)CC2CC(NC(C3(C)CCOCC3)=O)C(C2)C1 N1(C(C=Cc2c(C)ncs2)=O)CCCC2(C1)CN(C(c1ccc(CO)cn1)=O)C2 Cc1cc(C)n2nc(C(=O)NC3CC4CC3N(C(=O)CNC=O)C4)cc2n1 Cc1cc2sc(C(N3CC4C(CN(C)C(C5CCNC(=O)C5)=O)C4C3)=O)cc2s1 C1(OC)CN(C(C2CC2C#N)=O)CC1NC(c1ccc(-c2ccccc2F)[nH]1)=O C1(NC(COC(C)=O)=O)CN(C(=O)Cn2[nH]cnc2=N)CC1C N12C3CCC1CN(C3)C(=O)c1c(nc(OC)s1)CC2=O.c1(S)ccccc1.CO C1(C(N(CCC(C)(C)F)C)=O)Cc2ccccc2N1C c1(C2CC(=O)NCC2)ccc(NC(C2CCCN(C(C3(O)CCC3)=O)C2)=O)cc1 N1(CCC(N2CCC(CCNC(C(C)C3CC3)=O)C2)=O)CCP(C)(=O)CC1 c1(NC(C2(COC)CC2)=O)cc(CCO)ccc1Cl.c12ccc(cn1)NC2 c1(C(N(C(CSC)C)C)=O)cn(CCNC(C2SCC=C2C)=O)nn1 C(=O)(CC(CC1CC1)NC(c1ccc(CO)cc1)=O)NCC(CC)(C)OC C#Cc1cc(F)ccc1CNC1CCCC(C(=O)Nc2ccc(Br)c(C)c2C)C1 CC1(C(N2CC(NC(=O)COCCCF)C(O)C2)=O)CC2(CC2)C1 C(=O)(C(C(C)C)OC)N1CC(OC(=O)OC)C1.N1(C(C(=O)NCC)C)CCCCC1 C1(NC(C2(OCCC(=O)N3CCC3)CC2)=O)CCCC(C2CC2)C1 Cc1ccc2oc(C(=O)NC3CC3CNC(c3cn4cccnc4n3)=O)cc2c1 Cc1cc(Cl)nc(COC(=O)CN2CCN(CC(F)(F)F)S2(=O)=O)n1 C1(NC(CC2CCN(C)C2)=O)CC2(CCN(C(c3nc(Cl)cs3)=O)CC2)C1 C1(OC)CC(NC(=O)C=Cc2ccsc2)CN(C(C2CCCC(C)(C)C2)=O)C1 C(CC(C)C)(C(=O)NC(C)C(C)NC(=O)Cc1cc(C)cc(F)c1)NC(C)=O C(=O)(CCCN=C(NC(C)(C)C)NC(C)COC(C)C)OCCC c1(C(=O)NC23C(CN(C(C(C(=O)OCC)CC)=O)C2)C3)cc2c(nn1)CCOC2 CC1(C)CCC(C(=O)NCc2nc(CNC(C3CC=CC3)=O)cs2)C1 C1(C(=O)NC2CCCC(NC(CN(S(C)(=O)=O)C)=O)C2)CSC2(C)CCC(=O)N12 C1(C)(NC(c2ncn(CCNC(C(CN(C)C)O)=O)c2)=O)CCOC1=O CC1(C(=O)NCCC2CCCCC2)CC(O)CN1C(=O)C1=CCCCC1 N1(C(CNC(C2CCC(C)O2)=O)=O)CCC(O)C1C c1(CC(=O)N(C2CCCC(NC(=O)CC3OCCCO3)C2)C)ccnc(O)c1 N1(C(c2ocnc2C(F)F)=O)CC2CN(C(C3CC4(CCC4)CO3)=O)CC2C1 N1(C(CC2N(C)CCOC2)=O)CC(NC(c2cccnc2F)=O)C2CCCC2C1 N1(C(C23N(C(c4nccc(CC)c4)=O)CCC2C3)=O)C2CCC1COC2 N1(C(CN(C(C)C)C)=O)CCC2(C1)CN(C(=O)CCc1ncc[nH]1)CCO2 n1(CC)ccc(C(=O)NC2CCCCC2CNC(=O)CCOC)cc1=O c1(C(=O)NC2C3(CC(NC(c4nn(C)c(CO)c4)=O)C3)C2)n[nH]c2c1CCCC2 c1(C(=O)NCc2c(C(=O)NCC3N(C)CC(O)C3)con2)c[nH]c2ccncc12 N1(C(C(CCOCC)O)=O)CC2(CC(NC(C3CN(C(N)=O)C3)=O)CO2)C1 c1(NC(C(CCNC(c2ccccc2)C(C)C)O)=O)ccc2cnccc2c1 N1(C(c2c(OCC)snc2C)=O)CCC(NC(C23CSC(C2)C3)=O)CC(O)C1 C1(O)(CNC(=O)C=CC=C(Cl)Cl)CCN(C(C2CC(O)C2)=O)C1 c1(NC(C(C(C)C)C)CNC(c2cnn3c2OCCC3)=O)ncn(C)c(=O)c1Br N1(C(C2(CC#N)CC2)=O)CCCN(C(C2CC2c2ccccc2)=O)CCC1 c1(C(c2n(CCC(=O)OCC)nnn2)NCCC2(CC)CCC2)cc(C)c(Br)s1.CO n1(CC=C)cc(C(=O)N(C2CC2)CC2N(C(C3CCC(=O)N3)=O)CCC2)cn1 C1(CC(N2CCN(c3c(C#N)cncc3)CC2)=O)CCC2(CCOCC2)CO1 CC(C)CC(O)C(=O)N1C(C(=O)NC2(c3nn[nH]n3)CC2)CCC1C c1(CC(=O)NCCCNC(C2CCC(F)C2)=O)ccc(F)cn1 C1(F)(CNC(C(C)c2ccsc2)=O)CC(NC(=O)C(C)n2ccnc2)C1 C=Cc1cccc(CN2CCC(O)C(C(=O)NC(Cc3ccccc3)CO)C2)c1 C1(C(N(C)Cc2cnn(C)c2)=O)COC2(CCCC2)C1 C(=O)(C1=CCCNCC1)Nc1ccc(NC(CC)=O)c(C(C)C)c1 C12(CC(=O)N(C)CC3CC(F)CN3C(c3cc(Cl)n(C)n3)=O)COC(C)(C1)C2 C1(C(N2CC(NC(c3[nH]cc(C(N)=O)c3)=O)C2)=O)CCCN(CC(F)(F)F)C1 CC(=O)CCCCC(=O)NC1CCCCCN(C(c2ccnc(C)c2C)=O)C1 Cc1ncc2ccc(C(=O)NCC3C4CCC3CN(C(=O)CCC(N)=O)C4)cn12 N1(C(C=CCCC(C)C)=O)CCC(C)N(C(=O)CC2CCCC23CC3)CC1 C=CCCCC(=O)NC(C)(CSC)C(=O)N1CCC(CN=[N+]=[N-])C1 Cc1cc(Br)cc(F)c1C(=O)NCCN(C(=O)Cn1cnnc1O)C C=CCCCC(C)NC(c1ccc(CNC(=O)C(C)(C)n2cncn2)o1)=O CCCC(CNC(=O)C(CC1CCC1)NC(C1CCC2(CC1)CC2)=O)CCC c1(OCCN(C(C(=O)NCC(c2cccnc2)C)=O)C)ccccc1Br C1(CC(=O)NC2CCN(CCC)C2)CCCN(C(=O)C=Cc2cscn2)C1 C1(C(N2CC(CC(C)NC(CCC#CC)=O)C2)=O)CCc2nnc(C3CC3)n2C1 N1(C(CC2(CSC)CC2)=O)CC(NC(=O)CSCCC(C)C)CC12CCCCC2 c1(C(=O)NC(C(=O)N2C(C)CCC2)CCOCCO)cnn2c1OCC2 C=C(C)CC(C)C(=O)N1CCC(NC(c2ccc(C(=O)COC)cc2)=O)CC1C Cc1ccc(C(N2CCC(NC(c3ccnc(C(F)F)c3)=O)C(C)C2)=O)nc1C CC(C)(C)C(C(=O)NCC1CCCCCC1)NC(c1cc(O)cc(F)c1)=O c1(CC)cc(C)c(C(=O)NC2CCC(NC(=O)C(C)C3CCCC3)C2)o1 c1(C(=O)OC)cccn(CC(F)(F)F)c1=O.C1(=O)C(CC2CCCO2)N1 CC(C(=O)N1CCC(CNC(c2ccnc(OC(F)F)c2)=O)C1(C)C)S(N)(=O)=O CC(C)(C)C#CC(=O)N1CCN(C(c2ccncc2F)=O)C(CF)C1 Cc1cc(C)c(C(=O)NCC(C)(C2CCC2)NC(=O)CCC2CCCCO2)o1 CC1(C(N2CCN(C(=O)CCCCCF)C(C(F)F)C2)=O)CCCS1(=O)=O Cc1ccc(C(=O)N(C)C)c(C)c1Cl.N1(C(C(=O)N)=O)CCC(O)C1 N1(C(C(C)OC(C)C)=O)CCCC(n2cc(CN3CCOCC3)nn2)CC1 c1(-c2ccc(C(=O)NCC3(F)CC(NC(C4C(OC)C4)=O)C3)s2)cccc(F)c1 c1(-c2ccc(CN3CC(C)NC(=O)C3)c(F)c2)c[nH]c2ccccc12 C1(CNC(c2n[nH]c(C)c2F)=O)(NC(=O)CCn2cncn2)CCCCC1C C=CC(C)(C)CC(=O)NCCC(C)N(C(=O)CCCSC)C N1(C(C(C)=CC2CC2)=O)CCC(NC(C2CCCN(C(N)=O)C2)=O)C(O)C1 N1(CCN(C(c2cccc(OCCC)c2)=O)C)c2ccccc2CC1C c1(C(C)C)cccc(C(N2CC(NC(=O)C(F)CC3CCC3)C(C)C2)=O)c1 c1(CC(=O)NC2CN(C)C(=O)C2)ccc2c(c1)CCOC2 N1(C(c2ccc(C(OC)OC)o2)=O)CC(NC(c2snnc2C(C)C)=O)C2CC12 CCC(Cc1ccc(N)cc1)C(=O)NC1CCN(c2ccccc2)C1 N1(C(C2(OCN(C(CNC(=O)OC)=O)C)CC2)=O)CCCC2CCCCC12 C12(C(=O)NC(C)(C)CCNC(C3CCOCC34CCC4)=O)CCCN(CCC1)C2 C1(NCC2CCOC2)CCC(C(=O)NC(=O)CSCCCc2ccccn2)CC1 c1(OCC#N)ccccc1NCc1cnc(-c2ccccc2)s1 N1(C(C2CC2)=O)CCCC2COCC12.N12CCCC1NC(=O)C2=O N1(C(C(CSC)(C)C)=O)CCC(CO)C(NC(c2cnc(C3CC3)o2)=O)C1 c1(C(=O)NCC2C(NC(C(C)=CC)=O)C2)ccc(OC)c(Cl)c1OC N1(C(C=NOC)=O)CCC(NC(=O)C2=NOC(C(C)(C)C)C2)C(CO)CC1 Cc1ccc(C(N2CCC(NC(=O)CC34CCCC3C4)C(C(N)=O)C2)=O)nc1C C(N=c1[nH]c2c(c(=NC(C)C)[nH]1)CCCC2)c1n(CCC)nnn1 c1(N2CCC=C(C)C2)nc(N2CC(C(F)(F)F)OC(C)C2)c2c(n1)CCS2 CN1C(=O)CCC1C(=O)NCCC1(C(=O)NCC2(C)CCCN2C)CC1 C1(NC(c2ccc(CC)cc2)=O)CCN(C(C2CCCN2C)=O)CC1F C1(NC(CCOc2ccc(C)cc2)=O)CC2CCC(C1)N2C(=O)C(C#N)C1CC1 N1(C(c2c(C)onc2)=O)CCOCC1CN(C(=O)CC1CCC2CC12)C CCC(C)(C)CC(=O)NCC1C=CCN1C(=O)CCCc1nc(C(C)C)no1 C(=O)(CN=S(C)(C)=O)NCC(c1ccc(N(C)C)cc1)NC(Cn1c(C)ncc1)=O c1(N(CC=C)C)ncccc1S(=O)(=O)N1CCCC(N(C)C)CC1 N1(C(C(C(CC)O)C)=O)CCC(C2CCCN(C(=O)C3=CCC3)C2)CC1 Cc1c(Br)c(C(N2CCC(C(C)NC(C3CCOC3)=O)CC2)=O)nn1C c1(C(=O)NC(CCCC)CNC(=O)C(C)(C)CC)cc(OC)ncc1[N+](=O)[O-] C(=O)(CC(C)CC(C)C)N(C(CNC(c1cc(C)c(Cl)cc1)=O)C)C c1(CC(=O)N(CCCCNC(=O)COC2CCC2)C)c(F)cccc1Br C1(O)(CN(C)C(C2CC(=O)N(O)C2)=O)CCCN(C(=O)C(C)(C)C2CCC2)C1 N1(C(c2c(CC)noc2)=O)CCC2CN(C(=O)CS(=O)(=O)CC)CCC2C1 N1(C(c2nc(CCC)oc2)=O)CCC(C(F)(F)F)C(CNC(=O)C(C)(F)F)C1 c1(C(C(N2CCC(CC(C)C)C2)=O)N)cccc(I)c1 C1CCC(C2CCN(CC3C4CCC34)C2)C1 C=CCC(CNC(C1(CNC(=O)COC2CCC2)CC12CCC2)=O)CC(C)C C1(C(=O)NCCN(C)C(C2(C(N)=O)CC2)=O)CC(C(F)(F)F)CO1 c1(C(N2CCN(C)CC2C(N)=O)=O)ccc2c(c1)C(C)(C)CO2 C1(N(C(CCC)C)C(=O)C(C)OC(C)=O)CCC12CCNCC2 C(CC(=O)NCC1CC2(CCC2)C1)(CC(C)C)NC(C(C)N(CC)CC)=O C=Cn1nccc1C(N1CC(CNC(c2ccnc(OCC)c2)=O)C1)=O c1(C(=O)NC2CC(C)(NC(CC(c3ccccc3F)C)=O)C2)ccc(C#N)cc1 n1(CC)cc(I)c(C(N2CCC(c3cnco3)C2)C(=O)NCC(C)C)n1 CCCCC(C)CCC(=O)N1CCN(C(C23CCC(N(C)C)(CC2)CC3)=O)CC1 Cc1cc(C(=O)NCCCN2CCCC2)ncc1-c1nc(C)c(C)s1 C(=O)(CCCC(=O)N1CCC(NC(=O)C=C2CCCCC2(C)C)C(O)C1)OC CCC(C(=O)NCCCCC(C)NC(c1cnc(C)[nH]1)=O)C(C)C c1(NC(c2c(-n3ncc(C)c3)cncn2)=O)ccc(N2CCCC2)cc1F C1(CCC)CN(C(=O)C(CC)C(C)C)CCN1C(=O)C=C(C)c1cccs1 O=C(NNC(=O)C(O)c1ccncc1)c1cccc2[nH]ncc12 C(=O)(C(=O)C(C)(C)C)N1C(C(=O)NCC(CCC)(C)O)C=CC1 c1(OC)cc(C=O)ccc1O.c1(C(CN)=O)ccc(C(N)=O)cc1.C1CCO1 c1(C(N2CC(CC)C(NC(=O)C=CC(=O)N(C)C)CC2)=O)c(C)cc(C)cc1N c1(C(=O)Nc2cc(C)nc(C)c2C(=O)O)cccc(Cl)c1N=[N+]=[N-] C1(C(N(CCCCC)C)=O)C=CCN(C(=O)C(F)C(=O)OCC)C1 C(C(CC1CCCC1)C(=O)N1CCC(CC(F)F)C1)NC(CSC)=O CCC(C)CC(C(=O)NCC1(CC(=O)OC)CC1)NC(c1sccc1C)=O C12(NC(c3ccc(NC)cc3)=O)CCC1CN(C(c1ccc(CCF)cc1)=O)C2 c1(OC)cc2ccc(F)cc2nc1NS(=O)(=O)c1cc(-c2cccc(Cl)c2)n[nH]1 N1(C(c2c(CC)csc2)=O)CC(CC(=O)NC(c2coc(C(N)=O)c2)=O)CC1(C)C C1(CCNC(CCc2c(C)ncs2)=O)CN(C(=O)CC23CCC(CC2)C3)CCO1 N1(C(C(CCOC)C)=O)CCN(C(c2cnn(CC(C)C)c2N)=O)C(CCO)C1 C(=O)(CCCCC(C)(C)C)NC1(CCNC(c2cc(C(CC)C)c(C)o2)=O)CC1 c1(N2C(CNC(C(C)=C3CCCC3)=O)C(C)CC2)nc2ccccc2s1 N1(C(CC)=O)CCC2(CC1)CN(C(=O)CNC(C1CCC(C)CC1)=O)CC(C)O2 Cc1cc(Br)cnc1C(=O)N(CC(O)CNC(=O)CN1CC2CC2C1)C C12(C(=O)NC(=O)OC(C)(C)C)CC(Nc3ccccc3)(C1)C2 C(c1ccc([N+](=O)[O-])s1)=CC(N1C(CCNC(CSCC#C)=O)CCCC1)=O CC1=CCC(C(N2CCC(C)(NC(=O)Cc3ccc(C(F)(F)F)cc3)C2)=O)CC1 N1(C(C(N2CCC(OC)CC2)=O)=O)CC(=O)NC2CCCC2(C)C1 c1(C(N2C(CNC(CC(=C=C)C)=O)COCC2)=O)ccnc2cc(OC)ccc12 C=C1CCN(C(=O)CC2CCOCC2)C(C(N2CC(CC)C2)=O)C1 c1(C(N2C(C(C)NC(=O)Cc3cccs3)CCCC2)=O)ccc(Cl)c(Cl)c1O C1(C(=O)NCC2CN(C(C)C)C2)CC(F)CCN1C(=O)CC(O)CN(C)C C(=O)(CCCC(F)(F)F)N1C2C(C(=O)N(C(C(F)(F)F)C3CC3)CCO)C(C2)C1 C1(CC(=O)N(CCCN(C(=O)Cc2nc[nH]n2)C)C)CCCS(=O)(=O)C1 N1(C(Cc2ccc(C)c(O)c2)=O)CC2C=CC1C(C(=O)NCc1nc(=O)o[nH]1)C2 c1(C(N2CC(CCNC(=O)CCCC3CC3C)(OC)C2)=O)cc(C)cc(C#N)c1 CC1OC2CCC1(C(N1C(C(N3CCC(OCCF)C3)=O)CC3CC13)=O)C2 N1(C(=O)C=Cc2cocn2)CC2(CCC2)CC1CNC(C12COC(CCO1)C2)=O c1(NC2CCCCC2C(=O)NC(COC)C(C)C)ccc(C#N)c(C)n1 C1(CNC(=O)COCC(F)(F)F)CC2CCC1N2C(C1CC2CCC1CC2)=O Cc1oc(C2CC2)nc1C(N1CC(CNC(C2(C)CSC2)=O)C(C)C1)=O CN1CCCC(CC(=O)NCc2cccc(C(=O)N(C)CCN3CCCC3=O)c2)C1 N1(C(C(c2cccnc2)NC)=O)CCCCC12CCCNC2 c1(CC)nn(C)c(NCC(C2CC2)NC(c2ccc(Br)o2)=O)c1[N+](=O)[O-] C1(C(N)=O)CCCN(CCC(N2CC(NC(=O)COCCF)CC2CO)=O)C1 Cc1nnc2c(C(=O)NC3CC(NC(c4cccc5c4OCO5)=O)C3)nccn12 c1(NC(CSCC2C(C)(C)C2C#N)=O)ccc2c(c1)NC(=O)CC2 C1(NC(C2CNC(=O)N2)=O)(CO)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 c1(C(N2CCCC(O)(CCNC(C(C)CO)=O)C2)=O)nc2ccccc2nc1O C(=O)(C1=CC2C=CC1C2)NC(C(CC)C)C(=O)N1CC2CC1C1CC21 N#Cc1ccc(CCC(=O)NC2CCOCC2NC(C2CCC2)=O)c(F)c1 CC1(C)CCN(C(=O)C=Cc2ccco2)C1CNC(=O)CCc1ccncn1 c1(C2N(CC)CCC2)cc(C)c(Cl)cc1OC(C1OCCN(C)C1)=O.OC c1(C(N2CC3(C(NC(C(C)N(C)C)=O)CCS3)C2)=O)noc2c(F)cccc12 Cc1nc(C)c(C(=O)NC2(C(=O)Nc3cnsc3)CSC2)[nH]1 N=c1ccc(C(N2CC(O)(CCNC(=O)CC(O)C3CC3)C2)=O)n[nH]1 C#CCCCCC(=O)N1CCOC(CN(C)C(c2cccc(F)c2)=O)C1 CCCC(CC)(c1nnnn1CCCSC)NCc1ccc(CCCC)cc1 Cc1nc(C(N2CCN(CCN(C)C(C3CC4CCC34)=O)CC2)=O)c(C)n1C N1(CC)CCC(N(c2cnccn2)C(C)C)C1 c1(C(=O)NCC2(NC(C3C=C(C)CS3)=O)CCCCC2C)ccc2c(c1)NCC2 C1(Nc2ncnc(=N)[nH]2)CC(NC(C2=NOCC2)OC(C)C)C12CCOCC2 c1(CC(C)NC(=O)C=CCO)cncs1.C1(=O)CC2(CC2)N1 N1(C(C(COC)O)=O)CC2(CCCC(CNC(c3ncc(C)[nH]3)=O)O2)C1 n1(CCC=C)nc(-c2ccco2)nc1-c1ccc(OCOC)cc1 c1(C(N2C3C(N(C(c4c(C)cno4)=O)C)CC(C3)C2)=O)cn2cccc(F)c2n1 C1(NC(Cc2ccc(C)s2)=O)CC1C1CCCN(C(c2cccs2)=O)C1 C=CC(C)(CC)C(=O)N(CC(C)NC(c1cc(-c2ccncc2)[nH]n1)=O)C c1(N(CCCOCC=C)C)[nH]c(=NCC(C2CC2)C2CC2)nc2c1ncn2C CCCS(=O)(=O)CC(=O)NC1CCN(C(C2CCN2CC)=O)CC(O)C1 Cc1cccc(OCCC(=O)NC2CC2NC(=O)CN(C2CCC2)C)c1 C1(C(=O)NCC(C)CN(C)C(C2CN(C3CCOC3)C2)=O)(OC)CCCOC1 c1(CC(=O)N(C2CCCN(C(c3cc(C)no3)=O)C2)C)ccnc(F)c1F c1(C(=O)NCC(CC)NC(c2ccc(COC)o2)=O)ccn2ccsc12 c1(C(CC(=O)NCCCN(C(=O)CC2(C)CC2(F)F)C)C)c[nH]c2ccccc12 c1(OC(c2cccc(Oc3ccc(Br)nc3O)c2)=O)ncc(Cl)cc1Cl c1(C(=O)NCC(CC)NC(c2ccnc(C)n2)=O)csc2cc(OC)ccc12 O(NC(=O)C(O)C1CCCC1)CC(=O)NC1CCCN1C1CC1 N1(C(C=CC(N)=O)=O)CCC(C2CCCCN2C(C2CC=CCO2)=O)CC1 CCC(CCNC(C1(CC(C)C)CCNC1=O)=O)C(=O)N(C)CCOCCSC S(=O)(=O)(c1c[nH]c(C(=O)NC(C)CN(C)C(C2(C(C)(C)O)CCC2)=O)c1)NC CC(C)C(N=[N+]=[N-])C(=O)NC(C)CC(=O)NCC1CC(C)(C)CCO1 N1(C(c2c(CC)nn[nH]2)=O)CCCN(C(=O)CC(C)O)C(CO)C1 N1(C(c2c(C)n[nH]c2)=O)CCCC2(C1)CN(C(C1CC3C(C1)C3(F)F)=O)CCO2 c1(OC)cnoc1C(c1nnnn1CC1CCOCC1)NC1CCCC1 c1(OC)ccc(C(=O)NC2CN(C(C3(C(=O)O)CCCOC3)=O)CC2F)cc1 C1(NC(c2n(C)cnc2)=O)CC2CCC1N(C(c1cccc3c[nH]nc13)=O)C2 CN1CC(C(=O)NC(C2(O)CCCCC2)C(=O)NC2CC3C=CC2C3)CCC1=O C1(C(=O)NCc2cccc(C3(F)CNC3)c2)CCCC12OCCO2 C(c1cncnc1O)=CC(=O)NC1C(CNC(C(=Cc2ccccc2)OC)=O)C1 N1(C(c2c(C)coc2)=O)CCN(C)CC1CNC(c1cccc(N)c1O)=O N1(C(CCc2cnc(C)o2)=O)CCC=CC1C(=O)N(C)Cc1scnc1C c1(CC(N2CC(NC(CC(C)CN(C)C)=O)C(F)CC2)=O)c[nH]c2ccncc12 c1(C(=O)NCCC(=C)CNC(=O)C(C2CCCCC2)F)cn(C(C)C)nc1CC C1(CNC(C(C)C(C)O)=O)CN(C(=O)CC2CC3(CCC3)C2)CC(C)(C)C1 C1(CCNC(C2(Br)CC2(F)F)=O)CCN(C(=O)CC2CCCCC2)C1 c1(C(=O)NCC(C2CC2)NC(c2nc(C)oc2)=O)cc2n(n1)CCCC2O c1(-c2ccn(C)n2)cccc(CN2CCC(C(N3CCCC(Br)C3)=O)CC2)c1 C=C(C)CC(C(=O)NC(CNC(c1cc(N)cc(F)c1)=O)CCCC)OC N1(C(C2CCCC(NC(c3c(C)nco3)=O)CC2)=O)CC2CC(O)CC2C1 C(C1(C)OCCc2sccc21)NC1CCCN(c2nc(C)cc(OC)n2)C1 CCCC(CC)CCC(=O)NC1N(C(C2CCC(C(=O)OC)CC2)=O)CC1(F)F Cc1nc2nccc(N3CCC(C)C(NC(c4cccc(C(N)=O)c4)=O)C3)n2n1 c1(C(N2CC3C(CNC(=O)CC4OCCO4)(C3)C2)=O)ccc(O)c2ccccc12 C1(NC(=O)Cc2scnc2-c2cccs2)CCCC(NC(c2n[nH]cc2F)=O)C1 Cc1cc(-c2cn(CCCN(C(=O)C(=Cc3ccccc3)C)C)nn2)cnc1F N1(C(CC(C=C)CC)=O)CC2CCC(C1)N2C(=O)CCCCCF C1(C(C)C(N2CCC(C(=O)NC3CCC(=O)O3)CC2)=O)CCCN(C(N)=O)C1 c1(C(=O)NC2CC(NC(=O)CC3CCC4CC34)C(O)C2)cc2n(n1)CCCC2 C1(CC(N2CCCC(N(CCO)C(C3CCOC3)=O)C2)=O)CN2CCC1CC2 C#CCC(CC#C)C(=O)N1CCC(NC(C2CCCSC2C)=O)C(CO)C1 Cc1ccc(O)c(C(N2CCOCC2CNC(=O)Cc2ccc(Cl)cc2Cl)=O)n1 Cc1ocnc1C(=O)NCc1cn(Cc2ccc(C(=O)O)o2)nn1 Cc1ccc(C=CC(N2CC(O)CC2CCc2cccs2)=O)cc1 c1(C(=O)Nc2cccc(C(CC)OC(C)(C)C)c2)cc(F)c(F)cc1N CC1(C(=O)NCCC23CCC2CN(C(=O)CCc2cccs2)C3)CCC(=O)NC1 c1(OC)cc(C)cc(CNC(=O)CCC2CC2CC)c1O.C12CN(C1)C(=O)CS2 C(=O)(C1=CCCC1(C)C)N1CC(C(C)C)N(C(=O)C(F)C2CCC2)CC1 C12(CNC(CCCOCC)=O)CCC(CC1)N2C(C1CC1c1ccccn1)=O C12(NC(Cc3ccc(OC)c(O)c3)=O)CCCC1CN(C(=O)CN1CC(C)C1)C2 C1(NC(CN(C(COC)=O)C)=O)CC(F)CN(C(C2(C)CCC(=O)NC2)=O)C1 C(=O)(C(F)(F)CC1CC1)NC1CCC(NC(C(CC)F)=O)C1 C(CCCC(=O)NN(CCCC(N1C(C)CCCC1)=O)C)N(C)CC.CC Cc1nc(-c2ccc(CN(C3CCC3)C)cc2)n(CCC(=O)OC(C)C)n1 N1(CCNC(CN(C(C)=O)C)=O)CCCN(C(C2CC2C2(C)COC2)=O)CC1 N1(C(CC2CC(C)C2)=O)CCC=CC1C(=O)Nc1ccc(N2CCCC2)cc1 c1(OC)ccc(C(N2CCN(CCN3CCOC3=O)CC2)=O)cc1Br Cc1c(C(=O)NC2(CCNC(c3ccc(=N)[nH]c3)=O)CC2)cnn1CC1CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(NC(C(C)SCC)=O)C2(C1)CCC2 N1(C(c2ccc(CO)cc2)=O)CC(CO)C2(C1)CN(C(C1CC3(CC3)C1)=O)C2 C(C(Cc1ccccc1)N=c1[nH]c2c(c(=NCC3(Br)CC3)[nH]1)CCCC2)OC C1(NC(c2coc(-c3ccccc3Cl)n2)=O)CC2CC1N(C(c1cscn1)=O)C2 c1(CC)nc(C)cc(=NC2CCN(C(c3cc(C)cc(Br)c3)=O)CC23CCC3)[nH]1 c1(C(N2C(C)C(NC(=O)C=Cc3cccs3)CCC2)=O)cc(F)cc(N)c1N c1(CC)ccc(C)c(NC(=O)C#CCNC(=O)CC2CCCC2C)c1 CCC(C)(COC)C(=O)N1CC(N(C(C2C=CCS2)=O)C)C2(CC2)C1 N1(C(C(CC)SC)=O)CC(CNC(=O)C(=O)NCC2CC2)C2(CCC2)C1 C1(NC(c2[nH]cc(C)c2)=O)CC(NC(c2occc2C2CC2)=O)C(O)C1 c1(CNC(C2(NC(COCCCCC)=O)CC2(C)C)=O)cccc(CC)n1 N1(C(Cc2c(C)con2)=O)CCN2CCN(C(=O)C=Cc3cn(C)cn3)CC2C1 C1(NC(C(c2cccc(F)c2)(C)C)=O)CCCC12CN(C(=O)CC1C=CCC1)C2 c1(C(=O)NC(CC=C)C)cc(CNC(C2(Cl)CC2C(C)=O)=O)ccn1 c1(CC(C(=O)NC2CC(C(C)NC(c3coc(Cl)n3)=O)C2)C)ccc(F)cc1 C1(C(N2C(COC)CC2)=O)CN(C(=O)CC(C)(C)C(C)=O)CC1C1CC1 C#Cc1cccc(C(=O)NCC2CN(C(=O)CC3OCCC3C)C2)c1F C(CCC(O)C(=O)NCc1cc(C2CC2)n[nH]1)NC(c1n[nH]c(C)c1Cl)=O C(=O)(CC(C)C(F)(F)F)N1CCC(C(N(C(C)CC2CC2)C)=O)(CF)C1 C1(C(N(CC=CC(=O)NCC(CC)OC)C)=O)(CC)CCOC1 N1(C(C(CCSC)O)=O)CCN(C(=O)C(C)(C)CO)CC1CF CC1C(NC(C2CN=C3N=CNN3C2)=O)CC2CCC1N2C(c1cn[nH]c1)=O C1(NC(c2nccc(C(N)=O)c2)=O)CN(C(c2cc3sccc3s2)=O)CCC1F Cc1cc(C(=O)NCC(C)CC(=O)NC(c2n[nH]c(C)n2)(C)C)n(C)n1 CC1C(CC(=O)O)CC(C)N1Cc1ccccc1N(C)NC(c1ccco1)=O CCC(C)CCCCC(=O)N1CC2CC1CN(C(=O)CC1CC=CC1)C2 N1(C(CC=C)=O)CC(NC(c2ccc(OC)o2)=O)CC12CCOC2 CC1CN(C(=O)C(C)Oc2ccccc2Cl)CC1(C)CNC(=O)C(F)=CCCF C1(NC(c2cnc(SC)[nH]2)=O)CC(NC(c2ccnc(O)c2)=O)C12CCC2 C1(NC(CCC(C)OC)=O)CN(C(c2cccc(Cl)c2F)=O)CC2CCCC12 Cc1cnc(C(N2CC(C(=O)OCC(F)(F)F)C2)=O)cc1Cl c1(CNC2C(CN)CCC2)nc2cc(Cl)ccc2s1.C1C(=O)O1 Cc1cccc(SCC(=O)NC2CN(C(C3CCCC3(F)F)=O)CC2C)c1 C1(C(N(C2CCN(C(C3CC(CC)C3)=O)CC2)CC#C)=O)CC(=O)N(C2CC2)C1 c1(C(=O)NCCC2(NC(CCc3cnc(C)s3)=O)CCC2)ccc2nncn2c1 C1(C#N)(C(=O)NC2CC(CNC(C3(CC=C)CC3)=O)C2)CC1C(F)(F)F C1(CNC(=O)CSCCC#N)C2CCC(C2)N1C(c1ccc(CO)o1)=O N1(C(CC)=O)CCCC1C(C)NC(=O)Cn1cccn1 N1(C(CN(C)CC)=O)CCN(C(=O)C=CSc2cccs2)CC1c1cccnc1 C1(C(N(CCCNC(COCCCCCC)=O)C)=O)CCCC(CSC)C1 c1(CNC(NOCCN(C)C)=O)ccnc(OC(F)F)c1 Cc1nc(O)nc(C)c1C(=O)NC(C)C(C)NC(C12COC(CF)(C1)C2)=O N1(C(=O)CCC2OCCO2)CCCCC1C1(NC(=O)CC2(O)CCOC2)CC1 c1(C(=O)NC23CCC(NC(Cc4c(C)nsc4)=O)(CC2)C3)ccc(S(C)(=O)=O)s1 C1(C(=O)NCCN(C)C(c2cncn2C2CC2)=O)OC(C)(C)OC1(C)C CC(C)CC(C)CC(=O)N1CCC=C(C(=O)N2CCOCC(C)(C)C2)C1 C(=O)(CCCC(=O)N(CC(C)CNC(=O)CCc1ccncc1)C)N(CC)CC C(=O)(C(C(C)CC(C)C)N1CC2CCOC2C1)NC c1(NC(N(C(C)(C)C(C)N2CCOCC2)C)=O)cccc(OCC(F)(F)F)n1 N1(C(CC=CCC)=O)CCCC(CNC(c2cc(F)nc(F)c2)=O)CC1 C12(NCCCCNCc3ccncc3)COCC(C1)C2 c1(C(N2CCOCC(NC(C(CC=CCC)C)=O)C2)=O)ccc(OC)c(Cl)c1F N1(C(C=NOC)=O)CC2CCCCC2(CNC(c2cc(Cl)ccc2NC)=O)C1 N1(C(C2(NC(c3c(C)occ3)=O)CCSC2)=O)CCc2nnnn2CC1 Cc1nc(=NCC2C3CN(C(=O)CNC(C4CCCCC4)=O)CC23)[nH]cc1[N+](=O)[O-] c1(NC(C)=O)ccc(N(C)CC2COC(=O)C2)cc1F C1(NC(CC=C(C)C)=O)CCC(NC(c2ccnn2C(F)F)=O)CC1 N1(C(CNC(CC)=O)=O)CCC2(CCCC2CNC(=O)C(C)(C)C(=O)OC)CC1 C12(C(N3C(C)CCC3)=O)CCC(CN(C(=O)C(C)OC(C)(C)C)C1)C2 N1(C(Cc2c(C)con2)=O)CC(C)CN(C(C2CCC(C)(C)C2)=O)C(C)C1 C(=O)(C(F)(CNC(c1cccnc1C1CC1)=O)C(C)C)NCC(CC)OC C1(NC(=O)NCC2(c3c(C)ccnc3)CC2)CCc2nnc(C(C)(C)C)n2C1 c1(C(N2CC3C(C(N4C(C#N)CCCC4)=O)C3C2)=O)ccc2sncc2c1 C(=O)(C(C)(C)CO)N1CCC(NC(C=C(C)C(C)(C)C)=O)C1 C1(CC=C)(C(=O)N(C2CCOC2)C)CN(C(=O)Cc2nocc2C)C1 N1(C(c2c(CCC)nco2)=O)CCC2(CC2)CC1C(=O)NC(C)CCCO Cc1nc2c(o1)CCCC2CC(=O)NCC1C=CCN1C(=O)C1CC1 C1(C(N(C)CCn2cnnc2)=O)CC(N=[N+]=[N-])CN1C(=O)CCn1cncn1 C(C(C)(C)C(=O)NC1CN(C(C2CC23CCC3)=O)CC1c1ccccc1)OC c1(CC(N2C(C3CCN(C(CC=CC)=O)C3)CCCC2)=O)cnn2c1CCCC2 C(c1cccc(F)c1)=CC(=O)NC1(CNC(Cc2n(C)ncc2N)=O)CCCC1 Cc1nc(C(C)C)ncc1C(=O)NCC1(C)CCCN1C(=O)CC(C)N(C)C C1(C(=O)NC2CCN(C(CCC)=O)CC2O)OC2CCCCC2C1C c1(C(=O)NCC2C(NC(CCN(C)CC)=O)CC2)nc(Cl)c(Cl)s1 O=C1CCC(C(=O)NCC(C2CC2)NC(C2CCCCC23CCC3)=O)=NN1 c1(N2CC(C)(C)C2)cccc(NS(=O)(=O)Cc2cccc(CC(=O)O)c2)c1 c1(NC(C2CCN(C(C(c3ccnn3C)C)=O)CC2)=O)cccc(C#N)c1 c1(OCC)ccccc1C(=O)NCC1CC1NC(=O)C=Cc1cnc[nH]1 c1(NCc2ccc(CC)cc2F)ccc(S(=O)(=O)NC2(C)CC2)cc1F C(CC(=O)C(C)(C)C)c1cn(C(C(=O)N(C(CCCC)C)C(C)C)C)nn1 C1(C(=O)NCc2n(CCC)ccn2)CC(NC(=O)CCc2ccco2)C1(C)C c1(C(C(=O)NCC(=C)C)N(C)CCOCC2CCOC2)ccnn1CC(C)C c1(C(N2CCCN(C(c3cc(C)ns3)=O)CC2C)=O)ccc2c(c1)nnn2C N1(C(CCC2C(C)C2)=O)CCC(C)N(C(=O)Nc2cnc(C3CC3)nc2C)CC1 N1(C(Cc2ccc(OC)cc2)=O)CCC2CN(C(=O)C(C)O)C(C)C12 C(=O)(C1=NOC(c2ccccc2)C1)N(CC(C)NC(c1ccc(COC)o1)=O)C C(CCCCC(=O)NC1CC2CC1N(C(=O)C(C)N=[N+]=[N-])C2)OC CCCC(C(=O)N1CC(OCC(=O)NC(CC)C(=O)OCC)C1)NC(N)=O c1(C(C)C(=O)NC2CC(NC(=O)CCNC(=O)C(C)(C)C)C2)c(Cl)cccc1Cl C12(COC)COC(C(=O)NCc3ccccc3SC(F)F)(C1)C2 O=S(=O)(c1c(F)cccc1F)N1CCOC(CNC(c2cc(Br)ccc2Br)=O)C1 c1(C(=O)NCCCCCn2cc(CCC3(OC)CCC3)nn2)cccc(C)c1F Cc1c(NCCc2ccccn2)ncnc1N1CCC(CC(=O)NC)CC1 c1(N2CC=C(CCNC(C3(C)CC3(F)Cl)=O)CC2)ncc(Br)cc1[N+](=O)[O-] C(=O)(CC(C)(C)CC(F)(F)F)N.n1(CC(=O)N(C)CCC2CC2)ccc(O)nc1=O C1(CNC(CN(C(=O)CCc2cccnc2)CC(C)C)=O)(CO)CCSC1 C1(C(=O)NCC(C2CC2)NC(C2(CC=C)CC2)=O)CCC2C(C1)C2(F)F C12(C(=O)NC3C(CNC(c4cnc[nH]4)=O)CC3)CCC(C(F)(F)F)(CC1)CC2 N1(C(=O)CCc2ccncn2)CCCC2(CNC(=O)C(F)(F)C(F)F)CCCC12 N1(C(c2c(C)c(F)ccc2)=O)CCC2CCN(C(=O)C(C)S(N)(=O)=O)C2C1 Cc1[nH]c(C#N)cc1COC(c1cc(C(F)(F)C(F)(F)F)on1)=O N1(C(C(CCC)C(C)C)=O)CCC2(CCCN2C(c2cc(=N)[nH]c(Cl)n2)=O)C1 Cc1c(C(=O)NCC2CN(C(=O)C(F)C(C)C)CC2(C)C)sc2cncn12 N1(C(c2c(C)cnnc2)=O)CCC(NC(C2CC(N(C)C)C2)=O)C(O)C1 c1(SC)nc(O)nc(C)c1C(=O)NCC(C)(C)CNC(=O)CCc1cnn[nH]1 c1(OC(C)C)cccc(C(N2CC3CC2CN3Cc2cnc(O)cc2O)=O)c1Cl N1(C(CCOCC#C)=O)CC2CCCC2(NC(=O)CCc2ccccc2C#N)C1 CC1(CNC(C2CCC3(CC2)CC3)=O)CCCN(C(=O)COC(F)(F)F)C1 c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(Cl)s2)ccn2ccnc2n1 c1(C(CO)NC(CN(C(=O)COCC2CCCC2)CCC)=O)ccco1 C1(C(=O)OC)C(O)CCN1C(=O)CC1(NC(=O)CC2CCCC3CC23)CC1 C(CC(C)C)(C(=O)NC1CC(=O)NC1=O)NC(c1c(C)cccn1)=O C(CO)(C(=O)NCC1(C(=O)NCC2CC=CCC2)CCC1)N(C)C C1(C(=O)Nc2nc(C)cc(C)n2)CC2(CC2)CN1C(=O)CSC1CCC(=O)NC1=O C(C(C(=O)NOC(C)CCC)C(C)(C)C)NC(c1cccc(C#C)c1C)=O N1(C(c2c(C)cc[nH]2)=O)CCCC12CCC(NC(C13CC(C1)C3)=O)CC2 c1(SC)c(C(=O)NC2CN(C(=O)CCCc3nncn3C)CC2C)cccc1F C1(OC)(CNC(C2CCCC2CNC(c2cc(OC)no2)=O)=O)CCCC1 CC12CN(C(C3CCCO3)=O)CC1CN(C(C1(c3cccs3)CCCC1)=O)C2 C(CCC(=O)NCC(C)NC(c1[nH]ccc1-c1ccccc1)=O)OC(C)C CCC(CC)(CO)C(=O)N(C1CCN(C(=O)Cc2cncn2C2CC2)CC1)C C(=O)(CS(=O)(=O)C(C)C)NC(C1CCN(C(c2c(C#N)cnn2C)=O)CC1)C c1(C(=O)NCCC2CN(C(c3[nH]n(C)c(=O)n3)=O)C2)ccc(F)c(C(F)F)c1 C(C)(C(=O)N(CCCO)OC)N(C(c1n[nH]c(CC)c1C)=O)C c1(OC)ccc2ncccc2c1C(=O)NCC1CC1CNC(c1csc(O)n1)=O C1(C(N(CC(C)NC(=O)C(N2CCCC2)C2CC2)C)=O)CCN(CC(F)F)CC1 C(CCC(N)=O)(C(=O)NC1CN(C(C2CC23CCC3)=O)CC1OC)NC(C)=O C(=O)(C(CC)CC)NC(CNC(CC=CCC)=O)C(C)C c1(C(=O)NCC2C(CNC(CCNS(CC)(=O)=O)=O)C2)ccc2c(c1)nc(C)n2C c1(CC(=O)NC(CNC(C2CC(C)(O)C2)=O)CO)cc(C(F)(F)F)c(O)nn1 C(c1ccc(F)cc1)=C(C)C(=O)N1CCC1CNC(C1CC12CC2)=O C(=O)(C1=CCCOC1)NCC(C)(CNC(C1CC(C)(C)CO1)=O)OC CCC1=C(C(=O)N(C2(O)CCN(C(=O)CSCCC(F)(F)F)C2)C)CCCO1 C(C)(CC(=O)N1CCC(CNC(C2CC(C)(C)C2)=O)C1)(C1CCC1)N(C)C C1(NC(CN(CC)CC)=O)COCCN(C(C2CC(F)(F)CN2C)=O)C1 CP(C)(=O)C(O)C(=O)NCCc1ocnc1CNC(C1CSC1)=O C(CCC1CC1)(C(=O)NC1CCN(CC)C1)NC(CCN(CCC)C)=O.C(=O)(O)NC N1(C(CN(C(C)C)C(C2C(C)C2C)=O)=O)CC(N(C)C)C1 c1(C(=O)NCCCCNC(C(C)OCC)=O)cccc(C)c1O C12(C(=O)NCC3C(C)CN(C(C45CC(CN4C4CC4)C5)=O)C3)CCC(CC1)CO2 c1(OC)cccc(C(N2CC(NC(C3CCC(=O)C3)=O)CC2C)=O)c1 C1(CNC(C(CC)N(C)C)=O)CN(C(C2(C)CC=CC2)=O)CC1C C1(CNC(c2nc(OCC)oc2)=O)C(C)CCCN1C(=O)C=C1CCSCC1 N1(C(C2(COC)CC=CC2)=O)CC(CC(=O)NCC2CC(SC)C2)C(C)C1 CC1(C)CCC=C(C(=O)NC2CC(CNc3ncnc4c3cnn4C(C)(C)C)C2)C1 c1(NC(C2CCN2Cc2cc(I)ccc2F)=O)cc(Cl)ccc1O c1(C(=O)NCCC)cccc(NC(=O)CN(C)Cc2nnc(S)o2)c1 C1(CNC(c2n(C)ccc2)=O)CC2(CC2)CN1C(c1cccn(C)c1=O)=O c1(C(=O)NCC2N(C(Cc3cn(C)nn3)=O)CC2)c(F)cncc1Cl CC(C)(CN=c1[nH]c(=NCc2cccc(N)n2)[nH]c2ccsc12)CC(F)(F)F c1(CC(=O)NC2C(NC(Cc3cc(C)sc3)=O)CCC2)nc(F)c(F)cc1F c1(OC)cccc(NCC(=O)OCC)c1.c1(C(=O)OCCSC)cnc[nH]c1=N C1(C(N2C(C(N3C(CCC#C)CCC3)=O)CC(F)C2)=O)CC(=O)C12CCC2 C(c1cc(Cl)ccc1Br)=CC(=O)Nc1ccc(N2CCCCCC2)cc1 CN1CC2CC1N(C(=O)C(C1CCCCC1)NC(=O)Cc1cc[nH]c1)C2 CC1(NC(C2COCCO2)=O)CN(C(C2C(c3ccccc3)C2(C)C)=O)C1 c1(C(=O)NCCCOCCN(C(=O)CS(N)(=O)=O)C)ccc(-n2cnnc2)cc1 C1(NC(c2c[nH]c(=N)s2)=O)CC2CCC1C(NC(=O)C1=CC(O)CCC1)C2 c1(C(=O)NCC(C2CCOC2)NC(C2(COC)CC2)=O)cnc2sc(C)nc2c1 C1(C(=O)NC(C)(C)CNC(C2(C(=O)OC)CC2C(F)(F)F)=O)(COC)CCCC1.SC C(CC(N=c1cc(CC(C)C)c2nc(C)sc2[nH]1)c1nnnn1C)SC c1(NC(C2N(C(C3CCC(OCC)CC3)=O)CC2)=O)ccc(NC(C)=O)cc1 C(=O)(C1=NOCC1)NCCCC(C)NC(C1(c2cccc(Cl)c2)CC1)=O N1(C(C=C(CC)C)=O)CC2OCCN(C(c3oc(C(F)F)cc3C)=O)C2C1 c1(C(N2CCCN(C(c3c(C)cno3)=O)CC2)=O)ccc(F)c2cccnc12 C1(C(=O)NCCNC(CCC2CCC(C)O2)=O)CCc2ncccc2C1 Nc1cc(C(=O)NC2CCCCCN(C(=O)CC3CCC(=O)N3)C2)cc(F)c1O c1(C(=O)NC(CCNC(c2cc(OC)nc(F)c2)=O)C)ccc2nc(O)sc2c1 C=CCCCC(C(=O)NC(C)CCCO)NC(=O)C=Cc1ccncn1 c1(C(=O)NCC2(COC)CCCN2C(c2csc(Cl)c2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(CCc2c(C)ncs2)=O)CCC2CC(C1)CN(C(C1C(C)C1(F)F)=O)C2 C1(NC(CCn2c(C)csc2=O)=O)C2CC1CN(C(C1(O)CCC1)=O)C2 N1(C(C2CC=C(C)CC2)=O)CCCC(CC(N2CC(F)(F)CC2C)=O)CC1 c1(CC)cnc(O)c(C(=O)NC2(CNC(C3CCC34CCCO4)=O)CC2)c1 Cc1ccc(Cl)c(C(N2CCC(F)C(NC(=O)CCC(C)(F)F)C2)=O)c1N c1(CNC(C(C2CCCN(C(=O)C(C3CC3)C3CC3)C2)C)=O)ccnc(F)c1 c1(C(=O)NC(C2N(C(c3c(CC)n(C)cc3)=O)CCC2)C)cc(S(N)(=O)=O)cs1 C(=O)(CCS(=O)(=O)c1ccccc1Cl)N1CCC(C)C1c1ccc(C(C)C)cc1 C1(F)(CNC(CN(S(C)(=O)=O)C)=O)CC(NC(=O)CCc2cncs2)C1 C(=O)(C#CC1CCCC1)NC1CC2CC(NC(C3C(C)C(=O)C3)=O)C1C2 N1(C(c2ccc(C(=O)OC)n2C)=O)CCCCCC1CNC(=O)C=CC1CCC1 O=C(N=c1ccn(Cc2cccc(Br)c2)[nH]1)c1ccc(Cl)o1 C1(C(C)NC(=O)COC2CC(F)(F)C2)CCCN(C(=O)Cc2ccnn2C)C1 C1(CC=C)(C(=O)NCCC2CC2C2CC2)CCN(C(=O)CC=CC)C1 c1(OC)ccccc1C(C)S.C(=O)(CCCc1ccccc1)C(=O)CN [N-]=[N+]=NC1CN(C(c2cccc3ccnn23)=O)CC1NC(C1(Cl)CC1(F)F)=O c1(CC(=O)NCC(C)(C)OCCNC(C2C(C)C2C)=O)csc(C(C)(C)C)n1 c1(CC(=O)NCC2CCCN(C(c3ccc(CF)cc3)=O)C2)cc(F)ccc1O c1(OC)ccc(N)c(C(=O)NCCN(C(=O)C(C)CN(C)C)CCCN(C)C)c1 C1(CNC(c2c(C)coc2C)=O)CC2(CCC2)CN1C(=O)C=CC1CCOCC1 C(=O)(CC(O)C(=O)N1CCC(O)(CNC(=O)CCc2ccoc2)C1)OC(C)(C)C N1(CCC(=O)N(CCNC(C2C(OCC)C2)=O)CC2CC2)C(=O)NC(C)(C)C1=O N1(C(CCC(=O)OC)=O)CCN(C(=O)CCCC(C)=O)C(CO)C1 c1(C(=O)NC(C)CCNC(c2cc3c(s2)CCC3)=O)cccn2[nH]c(=N)nc12 c1(C(=O)NC(CC=C)CNC(c2ccc(C#N)cc2)=O)nc2cnccc2s1 C1(C(=O)NCC2N(C(c3c(C)sc(O)n3)=O)CC2)CN=C2N=CNN2C1 C=C(C)CCCC(=O)N1CCC(NC(=O)CC(C)F)C1(C)C C1(N(C(CCC=C)=O)C)CCC(NC(c2cn(C)c(C(F)F)n2)=O)CC1 C1(CNC(c2c(C)noc2)=O)(CO)CCN(C(c2cc(C3(C)CC3)on2)=O)CC1 c1(C(=O)NC23CCCN(C(c4c(C)[nH]cc4)=O)CC2C3)cc2nccn2c(O)n1 CC(C)C(C(=O)NCC1CCC(NC(C2CCOC(=O)N2)=O)CC1)n1cncn1 C12(CCC)CN(C(C3CCOC(C(F)(F)F)C3)=O)CC(C(=O)O)(C1)C2 C1(C(=O)NOCCSC)(CC=C)CCN(CC23CC(C(=O)NCC)(C2)C3)C1 c1(C(=O)NCCCOCCNC(C2C(CC)C2)=O)n[nH]c2c1CCC(C)(C)C2 C(C1=CCCN(C)C1)NC(C1C(CC)CCN1C(c1ccc(C(N)=O)o1)=O)=O c1(C(N2CC3CN(c4ccc(C)cc4)C3C2)=O)cnc2[nH]ncc2c1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(C1)SCCC2NC(C1CCn2nnnc2C1)=O c1(NC(C=CC(C)C)=O)cccc2c1C1CN(C(C3CCCN(C)C3)=O)CC1O2 c1(CC)cnc(O)c(C(=O)NC2CC23CC(NC(c2ccc(O)nc2Cl)=O)C3)c1 c1(C(=O)NCCC(C)NC(CC(CCCCC)O)=O)ccnc2cc(F)cnc12 N1(C(c2cc(COC)on2)=O)CC2CC1CCC2NC(=O)CCc1ncc[nH]1 C1(NC(C2CN(CC)C(=O)C2)=O)CC2CC(C1)N(C(c1cc(O)no1)=O)C2 C1(C(=O)NCC=CCNC(c2c(C)cc(OC)nc2)=O)CN2CCN1CC2C C1(C(=O)NC23CC(NC(c4cn(C)[nH]c4=N)=O)(C2)C3)CC1C1CC(F)(F)C1 CN1CCn2nc(C(N3CCC(CN(C(=O)CC4CC(F)C4)C)CC3)=O)cc2C1 C12(C(N3CCC(O)(CNC(c4cn(CC=C)nc4)=O)C3)=O)CC1Cc1c[nH]nc12 C1(c2n(C3C(C)CCO3)nc(C3CCCC3)n2)C2Cc3ccccc3C12 C1(C(N2CC(O)(CNC(c3c(C)noc3C)=O)C2)=O)CCCC12NC(=O)NC2=O c1(OCC=C)cccc(C=C2SC(=S)NC=C2CC(CN)C(C)C)c1 C1(CNC(c2cnc(SC)nc2O)=O)CC2(CO1)CN(C(C1(C)CC1(F)Cl)=O)C2 C1(C(N(CCOC)CC)=O)C=CCN(C(C2CC(C)(CC)C2)=O)C1 N1(C(c2ccc(CCC)[nH]2)=O)CCC(NC(c2cccc(OC)c2)=O)C(O)C1 N1(C(c2c(C)cc(F)s2)=O)CCCC(NC(=O)CCc2nncn2C)C1C C#CCC(C)C(=O)N1CCCC(N2CCCC2=O)C1.C1(=O)CN1CC c1(NC(C(=O)NC(c2scc(C)n2)C)=O)cc(C#N)cn1C(C)C C1(N(C(CCOCCOC)=O)CCO)CCN(C(C2CCCO2)=O)C1 c1(C(N2C(C(C)C)C(NC(=O)C(C3CCOCC3)F)CC2)=O)cc(N)ccc1O C(=O)(C(O)(C(F)(F)F)C1CC1)N(C(C)CNC(c1cccnc1S)=O)C C(C(C)C(C)C(=O)NC1CC(C)(NC(c2ccc(CSC)o2)=O)C1)OC N1(C(c2c(OCC)ccc(Cl)n2)=O)CC(NC(C2CCO2)=O)C2(CCOCC2)C1 C1(NC(C2(c3cccc(OC)c3)CC2)=O)C2CCN(C(=O)C=C(Cl)Cl)C12 c1(C(=O)NC(c2nc[nH]n2)CO)ccc(CNC(c2ccnn2CCF)=O)nc1 c1(CC)ncccc1C(=O)NC12CC1CN(C(c1ccccc1SC)=O)C2 C12(CNC(=O)Cc3csnn3)CCC1CCN2C(c1ccc(Cl)s1)=O c1(C(=O)NC2C(NC(=O)CCN3C(=O)CCC3=O)CC2)cc2c([nH]1)CCOC2 Cc1noc(C)c1CN(C(=O)CSCCNC(=O)C(C(C)C)N(C)C)C C(=O)(C(C)CCCC)N1CCC(N(C(=O)C(C)c2cncs2)CC#C)CC1 c1(C(=O)NC2CN(C(Cn3c(C)ncc3)=O)CC2C)cnc(O)c2ccccc12 C(=O)(C(C)(C)c1cnn(C)c1)N(CC(C)NC(C1C(C(=O)OC)CC1)=O)C N1(C(CC2C(C)(C)C(O)C2)=O)CCCC(CCNC(C23CC4CC2C3C4)=O)CC1 N1(C(CSCC)=O)CCC(C(C)CNC(C2CC(N3CC(O)C3)C2)=O)CC1 Cc1c[nH]nc1C(N1CC(C)(NC(=O)C(C)N(CC(F)(F)F)C)C1)=O Cc1c(C(=O)N(C2CCCCC2)C(C2CCCO2)CC(C)C)cnc2ncnn12 CC1CC=C(C(=O)NCC2(NC(=O)C(C)N(C)C)CCCCC2)CC1 C1(C2CCN(C(c3c(Br)cnn3C)=O)CC2)(NC(CSCC#C)=O)CCC1 C1(NC(C=CC(=O)NC)=O)CCN(C(=O)CCC2(C)CC2)CC1C C(CC)(C(=O)NC1(C(=O)NCCSCC(C)C)CSC1)=CCCC C1(CNC(CC2(C)CCCO2)=O)CCN(C(c2cc(Br)n[nH]2)=O)CC1(F)F C1(CCNC(C2CN(C(C)C)C2)=O)CCCN(C(=O)CC2CSC2)CC1 c1(C(N2CC(CNC(C(CSC)C)=O)C(C)CC2)=O)cc2cccc(C)n2n1 C1(NC(C2(CNC(=O)Cn3cncn3)CC3(CC3)C2)=O)CC2CCC(C1)O2 CC1CN(C(=O)CSCc2cccnc2)CCC1NC(=O)Cn1cnc(C#N)n1 N1(C(c2cc(C(F)(F)F)ccc2Cl)=O)CCC2CN(C(c3cc(Cl)ns3)=O)C2C1 C(C(CC1CCCC1)C(=O)NCC(CO)N(C)C)NC(C1(CC)CC(=O)C1)=O C1(C(=O)NC2(CNC(=O)Cc3ccc(Cl)c(Cl)c3)CC2)CCN2CCOCC12 CCCC(C(=O)N1CCC(NC(c2cccc(OC)c2F)=O)C(O)C1)C(C)C c1(C(=O)OC)cnn2c1CC(CNC(c1ncn(C(C)(C)C)n1)=O)CC2 CC(C)CC(O)C(=O)N1C(C(N2CCCN(C3CC3)CC2)=O)CC2CC12 CN(C)NC(=O)CCC(=O)N1CCN(C(=O)CC#N)CC1c1cccnc1 c1(C(=O)NC(C(=O)NCC(CCCC)O)Cc2cn[nH]c2)cnc(C)c(C)c1 N1(C(CC(=O)OC)Cc2ccccc2Nc2ccccc2)CC(O)CC(C)(C)C1 O=C(CCCn1cccc1)NN1CCCC1C(=O)NCC(CO)C1CCC1 Cc1cc(C(=O)NC2CN(C(C3(C(C)(C)O)CC3)=O)CC2C)n(C)n1 C12(CNC(C3CCC(CC)O3)=O)CC1CN(C(=O)COCCCF)C2 N1(C(c2cc(C(N)=O)no2)=O)CC2CC(NC(=O)C3=CCCCC3)C1C2 CCCCCC(O)CC(=O)OC(C)(C)C.C12(CCC(C(F)F)C1)NC(=O)NC2 C1(Cc2n(CCC)nc(-c3ccoc3C)n2)CS(=O)(=O)c2ccccc2O1 Cc1ccc(C(=O)NC(C2CCOC2)CNC(c2c[nH]cc2Br)=O)s1 C1(C(=O)NCCC2CC(NC(C3CCSC3)=O)C2)CCCN1C(=O)C(F)(F)F c1(C(N2C3C(NC(C(CCCC)CC)=O)C(C3)C2C)=O)cccc2cnccc12 C1(c2n(C)ncc2)NC(=O)CCN(N2CCC(F)C(CO)C2)C1 c1(OCC)nccc(C(=O)NCC(CO)NC(=O)Cc2csc(S)n2)c1F N1(C(C(=O)NCC2(C)CCC2)=O)CCCC#CCC1 c1(C(=O)NCC2N(C(C(CCSC)O)=O)CCC2)cc(=O)c2ccc(F)cc2o1 Cc1cccc(SC(C)C)c1Cl.C123CC(C1)C(CO2)C(=O)N1CC(C1)NC3=O C1(F)(C(=O)NCc2ccc(CNC(CCC)=O)cc2)CS(=O)(=O)CC12CCC2 c1(CN2C(C(N3CCCCC3)=O)CCC(C(C)(C)C)C2)cccc2ncoc12 c1(C(=O)NC(C(C)NC(Cn2nc(C)c(Cl)c2)=O)C)ccc2c(c1)CNC(=O)N2 C12CCCCC1C(=O)NC2.c1(NC(CC2(COC)CC2)=O)cnn(C)c1.c1cn[nH]c1 C1(CC(=O)NC(CC)C2CC2)CN(C(=O)Nc2nn[nH]n2)C1 c1(CC)[nH]nc(Cl)c1C(=O)NCC1CN(C(=O)CCn2c(C)csc2=O)C1 c1(C(=O)OC)ccc2c(c1)N(C(CC(F)(Br)Br)=O)CCN2C C1(c2cn(Cc3ncon3)nn2)(NC(c2cc(SC)oc2)=O)CCCOC1 C(CN=C(NCC1(C(F)(F)F)CC1)NCC1CCCSC1)OC Cc1nc2ccc(F)c(CN3CCC(CC(=O)N(C)C(C)C)C3)c2[nH]1 CC1=C(C)CC(C(=O)NCC#CCNC(=O)CCc2cc(C)[nH]n2)CC1 C(=O)(C(C)(C)CCNC(=O)C1=CCSC1)NCc1c(COC)ocn1 c1(N2CCC(NC(c3n[nH]c(C)c3Cl)=O)C(C)C2)nc2cccnc2s1 C(C(CCNC(c1cn(C)nn1)=O)OC)NC(C1C(C(=O)OC)C1)=O C(C)(CO)(C(=O)NCCCSCCNC(=O)CCCc1cc(C)no1)NC(C)=O C1(C)(C(=O)NC2CC2)CCN(N(C)C)C1.c1(C(C(=O)OCC)N)c[nH]c(Br)c1 CCC(F)(F)C(C)(C)C(=O)NC1CN(C(c2cc(CF)on2)=O)CC1F C(C)(C)(CCC(=O)NC1CC1CNC(c1cn(CC(N)=O)nn1)=O)NC(C)=O CCC(C(=O)N1CCCCC1CNC(C1CC(OC(F)(F)F)C1)=O)C(C)O C1(NC(C(C)P(C)(C)=O)=O)CN(C(=O)COc2ccc(F)cc2Cl)CC1C1CC1 C#CCC(C)C(=O)N(CCCNC(=O)C(C)NC(C1CCOCC1)=O)C(C)C C(=O)(C1=C(Cl)CCCC1)NC(c1ccccc1)CNC(C1NC(=O)OC1)=O C(=O)(CC1=CCCCC1)NC1(CC(=O)N(CC(CC)CC)C2CC2)CC1 C(=O)(C(C)(C)CN(C)C(c1ccnc(O)c1)=O)NCC1(COC)CC1 N12CC(C)(C1)NC2=O.C(CC(C)C)SCC(=O)NC(=O)OC.C(CCOC)O C=CCCC(C)(C)C(=O)NCC1CCC1C(=O)NC(c1ccccc1)CO c1(SCC(=O)NCC(N(C(C(C)=CC2CC2)=O)C)C2CC2)ncccn1 Cc1nn(C)c(Cl)c1C(=O)N(CC(O)CN(C)C(C1OCC1(C)C)=O)C C(=O)(C1=C(C)C(C)(C)OC1=O)NCC(C)NC(COC1(C#C)COC1)=O C(=O)(C1CCCc2sc(=N)[nH]c21)NCCC(C)NC(c1c(C)nc(C)o1)=O N1(C(C2(CC#C)CCCC2)=O)CCCC(C(=O)NCCC2CC(F)C2)C1 NC(=O)CC(C1CC1)NC(C1CCCN1C(=O)CCCC1CCCO1)=O C(N=c1[nH]cnc2c1COC2)C1CN(C(C2CCC(C)C2)=O)CC1C CC(C)(CCC(=O)N1CC(NC(C2(C)CCCCO2)=O)C(C2CC2)C1)[N+](=O)[O-] C#Cc1cc(C(N2CC(NC(c3cccnn3)=O)CC(O)C2)=O)cc(Br)c1 N1(C(C(C)=C2CC2)=O)CCC(C2CC2)(CNC(c2ccnc(Cl)c2)=O)C1 c1(C(N2CC(NC(C3CCCCO3)=O)CC(C)(C)C2)=O)n[nH]c2c1CS(=O)(=O)C2 CC1CCN(C(c2ccc(Oc3cccc(Cl)c3Cl)nn2)=O)CC1O c1(C(N2CC(CNC(c3c(C)snn3)=O)C2)=O)coc2cc(F)ccc12 CC1CCC(NC(c2ccc(F)nc2)=O)CN1NC(C1CN(C(N)=O)C1)=O C#Cc1ccc(C(N2CCC(N(C(=O)CCSCCCC)CC)C(C)C2)=O)cc1 C1(NC(CCNC(C)=O)=O)CCCN(C(c2cn(C(C)(C)C)nc2C)=O)C1C c1(C(=O)NCCC(CNC(C=CC(C)(C)C)=O)O)cc(C#N)c[nH]1 C#CC1(C(=O)Nc2cnc(O)c(C)c2)CCN(C(c2ccn(C)c2)=O)C1 C1(C(=O)NC2(CNC(C(C)NC(CC)=O)=O)CC(F)(F)C2)CC2(COCCO2)C1 N1(C(CCC2(C)CC2)=O)C2CCC1CC(CNC(C1CC=CC(O)C1)=O)C2 Cc1c(C(=O)N(C(C)CCNC(=O)CNC(C2CCC2)=O)C)ccn1CC1CC1 O(N=C1CCCCCC1)CC(=O)NCCC1CC(NC(CC2CC(OC)C2)=O)C1 C1(C(N(C)CCOCCNC(C2CC(O)C2)=O)=O)CN(C)CC1c1ccccc1 N1(C(C(C)OCCCCCC)=O)CCC2CN(C(=O)Cc3cnn(C)c3C)C2C1 c1(SCCCCCC)ccc2oc(=O)c(-c3nc(C4CC4)nn3C3CC3)cc2c1 c1(OC)cc(C(=O)N(C2CCCN(C(=O)C(C)S(N)(=O)=O)C2)CC)c(O)c(Cl)c1 c1(C(=O)NCC2C(NC(c3ccc(C)cc3)=O)CCC2)ccc2c(n1)NCC2 C(=O)(C1=C(C)OCC1)N1CCC(N2CCN(C(C(C=C)O)=O)CC2)CC1 S(=O)(=O)(c1cc(C)cnc1NCC1(Nc2csc(COC)n2)CCC1)N(C)OC C1(C2CC2)(CNC(c2c(C)nc(C)o2)=O)CCN(C(=O)CC2C(=O)NN=C2C)C1 C1(C(=O)NCc2cc(CC)on2)N(C(=O)CN2CCSCC2)CCCC1(C)C Cc1c(NC)cccc1C(=O)NC1CC(NC(=O)CCC(C)(C)N(C)C)C1 CCC(CC(=O)NCC1CN(C(=O)CCOC2CCOCC2)CCCO1)C(C)C N=c1[nH]c2c(s1)CCCC2C(=O)NC1(CNC(c2cc3cc(Cl)ccc3[nH]2)=O)CC1 c1(C(=O)NC(CC(C)NC(c2c(C)ccn2C)=O)C)cc2c(nc1O)CCSC2 N(C(=NCCC(C)(F)F)NCc1ccc(C(C)(C)O)cc1)C(COC)C C(C)(C)(CCCNC(C1CCS(=O)(=O)C1)=O)NC(C=C(C)C(C)(C)C)=O C(=O)(C1=CCCCC1C)N(CCC(=O)NCC1CC(CC)C1)CC#C N1(C(C=CCC)=O)CC2CCCC2(NC(c2cc(C3CC3)n(CC)n2)=O)C1 CC(C)(F)CCC(=O)N1CC(NC(=O)CCc2cc(Cl)cs2)C2(CC2)C1 C(=O)(N=c1cc(-c2cccc(F)c2)[nH][nH]1)C1SCCN(C(C)=O)CC1 N1(C(c2cnc(OC)s2)=O)CC2CCOC2(CNC(c2cc(Cl)nnc2O)=O)C1 CC#CCCC(=O)N1CCC(N(CC(C)C)C(C2COCCO2)=O)CC1 c1(C(=O)OC)cc(NC(=O)NCCC(C)c2nc[nH]n2)ccn1 c1(C(=O)OCCN(CCOCC)CC)c(C)nn(CCC2CC2)c1Cl C#CCC(CC#C)C(=O)N1CCOCC1(C)c1cn(CC2CC2C(F)(F)F)nn1 c1(CNC(C2N(C(C3CC(CC)(CC)C3)=O)CCC2)=O)cc(F)c(F)cc1N C12(C(=O)NC(C)CC3CN(C(=O)CCC4CCC4)C3)CC1COC21CCC1 C1(CC)(CNC(c2coc(CNC(C3CC=CCO3)=O)n2)=O)CCCC1 c1(C(C)C)cc2c(NC3CC3NC(c3c(Cl)cccc3Cl)=O)ncnc2s1 c1(C(=O)NCC(C2CCN(C(=O)CCCC3CC3)C2)(C)O)cnc2scnc2c1 C1(CC)CC(C(=O)NC(C)CCCNC(=O)CSS(C)(=O)=O)CCO1 N1(C(c2cc(CCC)c(C)s2)=O)CC2CCCC2(NC(c2ccncn2)=O)C1 c1(CC(=O)NCCC(CNC(c2ccc(CCCCC)[nH]2)=O)O)cc(C)ccc1C N1(C(c2ccc(C)cc2)=O)CCN(C(c2cc(F)nc(F)c2)=O)CC1C(C)C N1(C(=O)Cn2cnnc2O)CCCOC(CNC(C2(c3ccccc3)CC2)=O)C1 C1(NC(CN2C(C)CC2)=O)CN(c2cc(Cl)nc(-c3ccccn3)n2)CC1(C)C Cc1ccc(N)c(C(=O)NCC=CCNC(c2csc(-c3ncccn3)n2)=O)c1 CC1CN(C(=O)C(C)(F)F)CC1NC(c1ccccc1OCc1ccccc1)=O C(=O)(C1=CCC(C)(C)CC1)N1CCC(CNC(C(CCOC)OC)=O)(OC)C1 CC1CCN(CC(=O)N(C)CCNC(C2C(c3ccccc3)C2(C)C)=O)C1 c1(Cc2cn(C(C)C)nn2)cc(C(F)(F)F)ccc1Cl.C12(OC)CCN(C1)C2 C1(C(=O)NC2CC(=O)N(CCN3CCNCC3)C2)CCCC12OCCO2 N1(CCC(=O)NCC23C(CN(C(C(C)S(N)(=O)=O)=O)C2)C3)Cc2ccccc2C1 N1(CCCC)CCC(C(=O)N(CC(C)NC(=O)CC2COCC(C)O2)C)CC1 Cc1ccc(C)n1CC(=O)NCCC1CCCCN1C(=O)COCC1CCCO1 c1(C(N(c2nc(OC)c(C)cn2)C2CC(N)C2)=O)cnc2cccnn12 CC1CC(CNC(=O)CC2OCCO2)CN1C(c1ccc(C(F)F)s1)=O C1(CNC(C(C(C)C)C2CCC2)=O)CN(C(C2CC2c2ccccc2)=O)CCCO1 Cc1nc2ncc(C(=O)NCC3(F)CCN(C(C4CC(C)(O)C4)=O)C3)c(=O)n2[nH]1 c1(C(N2C(C)CN(C(=O)Cn3cccc3)CC2)=O)cc2ncccc2s1 c1(OC)cc([N+](=O)[O-])c(NC(C2CN(C(c3cc(Cl)cc(Cl)c3Cl)=O)C2)=O)cc1C C1(CC#C)(C(=O)NC(C)(C)CCNC(=O)Cc2cccnc2NC)CCCCO1 c1(C(N2CC(NC(c3ccc(C4CC4)s3)=O)C(F)C2)=O)cnc2ccnn2c1 N1(C(C#CC)=O)CCC2C(OCCCCC(=O)NCCCOC)C2C1 CC1(C)CC(C(=O)NC2(C3CC3)CCN(C(c3cc4sccc4[nH]3)=O)C2)=NO1 CCCC(C(=O)NC1CCCN(C(C2(C3CCCO3)CC2)=O)C1)NC(C)=O n1(CC(=O)NC(C)CNC(=O)C=CC(=O)N(C)C)nc2n(c(=O)c1=O)CCOC2 c1(C(=O)NCC2(F)CC(NC(C(C=C=C)C)=O)C2)cccc(O)c1Br Cc1ccc(F)c(C(=O)NC2CC(NC(C3(C4CC4)CC3)=O)C2)n1 C1(NC(c2cnc(CC)[nH]2)=O)CCC(C)N(C(=O)CN(C)C(C)C)C1 c1(C(N2CCC(N(C(=O)CCc3ncccn3)CC3CC3)C2)=O)ncccc1O C1(N(C(c2n(CC)cc(Cl)c2)=O)C)CN(C(c2cc(N)cnc2C)=O)CC1(C)C c1(NC(CNC(C=Cc2n(CC)ccn2)=O)C(C)C)nccnc1C#N Cc1ncn(C)c(=O)c1C(=O)NCC12CC(CO1)N(C(=O)C(O)CC1CC1)C2 Cc1cc(C(=O)NC(C)CNC(c2ccc(F)c(CO)c2)=O)c2nn(C)cc2c1 c1(C(N2C(C)CC(NC(C(C(C)C)N(C)C)=O)C2)=O)cc(S(N)(=O)=O)co1 C12(F)CCCN(C1)C2.c1(CC)nc[nH]c1C(=O)Nc1ccn(COC)n1 Cc1ncccc1C(c1nnnn1C)NC(c1[nH]cnc1C(C)C)c1cccs1 N=S1(=O)CCN(C(c2cc(CNC(c3ccsc3Cl)=O)ccn2)=O)CC1 CC1CCC(=CC(=O)NCC(=C2CN(C(=O)COC3CCCC3)C2)F)C1 c1(C(=O)NC(CC=C)CNC(=O)Cc2[nH]cnc2C)cc2cc(C)ccc2o1 c1(C2CN(C(C(N3CCC(c4ccc(C)nc4)(O)C3)=O)=O)C2)cccc(Cl)c1F C1(c2nc(-c3n(CC)ncc3)nn2CC2CCCCO2)Cc2ccc(C)cc2S1 C1(C(=O)NCC2CN(C(C3(C(=O)NC)CCC3)=O)CC2O)CC2CCCC2C1 N1(C(c2cc(C)on2)=O)CCC2(CCN(C(c3cnccn3)=O)C2)C1 Cc1c(C(N2CCCC(NC(=O)CCc3ccc(=N)[nH]c3)C2)=O)cnn1CCO c1(C(=O)NCC23CC2CN(C(=O)C=Cc2cscn2)C3)cc2ncccc2[nH]1 c1(C(=O)NC2(C)CCN(C(C(C)OCC3CC3)=O)C2)cc2occc2[nH]1 c1(C(=O)NC2C(CNC(c3cccc(C)n3)=O)CCC2)cc(S(N)(=O)=O)cs1 CC1(C)CCC=C1C(=O)NC12CCCC1CN(C(=O)Cn1nnc(=N)[nH]1)C2 c1(C(=O)NC2C(CNC(C(c3scc(C)n3)C)=O)C2)cnc2ncnn2c1C Cc1cc(C(N2CC(NC(c3cscc3F)=O)C(C)C2)=O)c2cc(F)ccc2n1 C1(NC(C2C(OCC)CCCC2)=O)CCN(C(c2cccc(OC)c2)=O)CC1O CC1CC(CNC(c2cc(C3CC3)n(C)n2)=O)CN1C(=O)CN1CCC(F)CC1 C1(C(N(CCNC(C(C)(C)O)=O)C2CC2)=O)CCC2CCCCC2C1 c1(C(=O)Oc2ccc(CC#N)cc2)nc(-c2ccccc2)n2c1COCC2 n1(CC(=O)NC(CCNC(C(CC)(C)OC)=O)C)ccc(=O)c([N+](=O)[O-])c1 c1(C(=O)NCC(CNC(C2NC(=O)OC2C)=O)OC)[nH]nc([N+](=O)[O-])c1Cl C1(NCCS(=O)(=O)N(C)C)CC(O)CN(C(=O)CC(C)(C)C#N)C1 C12(C(N(CCC(=O)NCC(=O)NN=[N+]=[N-])CC#C)=O)CC(C)(CCO1)C2 Cc1ccnc(C)c1C(=O)N(C1CC1)CC1CCCN1C(C1CCC(=O)N(C)C1)=O C(=O)(CCC(CC)CC)NC1CN(C(C(CC#C)O)=O)CC(F)C1 c1(C(N2CCC3(NC(=O)COC4CCCCC4)C(C2)C3)=O)cccc2ccoc12 c1(CC)ccc(C(=O)NCC2CCN2C(C2CCSCC2)=O)c(C)c1 N(C)(S(=O)(=O)N(C)C)CC(N1CCC(N(CCOC)Cc2ccoc2Cl)CC1)=O c1(C(N2CC(O)(C(C(=O)NCCc3cccnc3)F)C2)=O)ncc2ccccn12 C1(CNC(C2C(OCC)CC2)=O)CCCCN(C(=O)CN(C)S(=O)(=O)N(C)C)C1 C1(NC(COc2cccc(CC)c2)=O)CCCC12CCCN(C(=O)C=CCO)C2 c1(C(=O)NCC2(CNC(c3cncnc3)=O)CC2)cccnc1NC1CC1 N1(C(c2c(CC)ncs2)=O)CCOCC(CCC(=O)NCCOC(C)=O)C1 CCCC(C)CC(=O)N1CC(C(=O)NC2CCCC(O)CC2)C(F)(F)C1 CC1CC(NC(c2cc(-c3ccn(C)c3)[nH]n2)=O)CN(C(c2cc[nH]n2)=O)C1 C1(C(=O)NCC(C2CCC2)OC(C)C)(CNC(COC)=O)CCCO1 N1(C(Cn2cccc(N)c2=O)=O)CC2(CCN(C(C3CC3C3CCCC3)=O)C2)C1 CCCC(CC(=O)NCc1cccnc1)NC(=O)COC(C)CC O=C(C1=CCN(C(=O)CC2=CCCC2)C1)NCC1CC2CCCC2C1 C(CC1CCC1)(C(=O)NCCSC)N(C(C(C1CC(OC)C1)F)=O)C1CCCC1 C(=O)(CCC(=O)C(C)(C)C)N1C(CO)CC(NC(C=CC(C)(C)SC)=O)C1 c1(C(N2CC(NC(COCCC)=O)C(CC3CC3)C2)=O)cc2n(c1)CCCC2 N1(C(C2(C)CCCC2)=O)CC2CN(C(C3CC4CCC3C4)=O)C2C1 c1(C(C)NC(C2(F)CC2)=O)ccc(CNC(=O)CC2(O)CCOC2)cc1 N1(C(N2CC(NC(=O)C3CC3)C2)=O)CCC(CNC(c2c(CC)noc2)=O)CC1 C1(CCNC(C2N(C(CN(C)C)=O)CCC=C2)=O)CCCCC12CC2 c1(CN(C(CC2CCN(C(CCNC(C)=O)=O)C2)=O)C)cccc(C)n1 C(CSC)(C(=O)NCC(C1CC1)NC(=O)CSc1csc(C)n1)OC N1(C(CNC(C)=O)=O)CC2C(CC(=O)Nc3cncc(C(F)F)c3)C2C1 O=C1Nc2cc(Cl)ccc2C1C1CCN(C(c2cc(Cl)c(F)c(Cl)c2)=O)CC1 C(=O)(CCCC(C)(C)C)NC(CCN(C(C=C(C)Cl)=O)C)C C=C(C)C(C)(C)C(=O)NCC1CN(C(=O)CCOc2cccnc2)C(C)(C)C1 N1(C(c2c(OC)ccnc2)=O)CCc2ccccc2C1CCNC(=O)CSC C1(C(=O)NCCCN(C(C2(CC=C)CC2)=O)C2CC2)Cc2nccnc2C1 Cn1nc(Br)cc1C(=O)COC(=O)CCC1CCCO1 C1(NC(C2N(CCC)CCC2)=O)CCC(C)(C)N(C(=O)C(F)C(F)(F)F)C1 N1(C(C)(C)C)CSCCSC1.C1(NCC#N)CCC12c1nnnn1C1CCC1S2 C1(NC(Cc2cn(CC)nc2)=O)CCN(C(C2CC(C)(C)C2)=O)C12CCCC2 c1(C(=O)NC2CN(C(CC3CCC(C)O3)=O)C2)cc(F)c(Cl)cc1F N1(C(c2cc(CC)c(C)s2)=O)CC(NC(c2cc(CCOC)on2)=O)CC(O)C1 Cc1cccn2cc(CCNC3CC4CCC3C4)nc12 c1(OC)cc(C(=O)N(C2CCC(NC(=O)CSCC(N)=O)C2)C)c(Cl)cc1Cl c1(C(=O)Nc2ccc(C(=O)Nc3ccc(C)c(Br)c3)nc2)c(Cl)cnc(Cl)c1Cl c1(C(C(=O)NCCN(C)C(C2NC(=O)C3CC23)=O)=O)c[nH]c2ccc(F)cc12 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(C)C)(C(=O)NCc2cnns2)CCC1 C(c1c(C)coc1C)=CC(=O)N(CCC(C(C)C)NC(c1c(C)cc(C)s1)=O)C C1(CNC(c2cc(O)no2)=O)CCCN1C(=O)CC1COC(=O)C1 c1(C(CNC(C2CC(NC(C3(CC(C)C)CCC3)=O)C2)=O)O)cnn(C)c1 O=C(C#CC1CCC1)NC1CCC1NC(=O)C(O)C(F)F CCCC(CC(C)C)C(=O)NCCC(O)CNC(c1oc(C2CC2)nc1C)=O c1(OCC=C)cc(F)ccc1C(=O)NC.c12nc(ncc1OC)N1CCN2CC1 c1(CC(N2CC3C(C(N4CCC(F)C4)=O)C3C2)=O)cc(F)ccc1[N+](=O)[O-] C12(CN(C(C(C#C)(C)C)=O)CC)CCCC1N(C(=O)CCC(C)(F)F)CCC2 Cc1ccc(C(=O)N(CC(C)CNC(=O)C2=CCCCC2)C)c(C)n1 c1(C(C)C(=O)NC(C)CCNC(=O)Cc2nccn2C)ccc(F)cc1 CS(=O)(=O)c1ccc(C=CC(=O)NC2CN(C(C3CC34CC4(F)F)=O)C2)o1 C1(CC)CCCC(NC(=O)CN2CCN(C)C(CF)C2)CC1.c1(O)ccc(SC)cc1 N1(C(c2ccc(CSCC)cc2)=O)CC(NC(C2CC3CC2CO3)=O)C(SC)C1 CC1CCOC(C(N2CC(CNC(C3(Cl)CC3)=O)C(C)C2)=O)C1 C12(C(N(C3CCOCC3N3CCOCC3)CC)=O)CC(C1)C(C)O2 N1(C(CCC2C(C)C2)=O)CCC(C2CC2)C1C(=O)NC1CCCCC1(F)F N1(CCC(=O)NCC2(NC(C3C4CNC(=O)C34)=O)CCOCC2)CCNC(=O)C1 [N-]=[N+]=NCC(C(=O)N1CC(SC(F)F)C1)NC(=O)C(O)CC1CC1 N1(C(C2CC=CC(O)C2)=O)CCC(C(=O)NOCC2CC3C=CC2C3)=C(F)C1 C(=O)(CCC(=O)NC1CC1)NCC(CN(C(=O)CCc1ccc(O)nc1)C)(C)C C1(C(=O)NCCCCCCNC(C(C)C(F)F)=O)Cc2nccnc2C1 c1(C(N2CCC(N(C(=O)CCCc3nccs3)C)C2)=O)nnc(O)nc1O n1(CCNC(c2c(C)con2)c2nnnn2C)cc(C(F)(F)F)ccc1=O N1(C(CC(C)=O)=O)CC2(CCN(C(C3(CC4CC4)CC3)=O)C2)C1 C1(C)(C(N2CCC(N(C(C(n3ncc(C)c3)C)=O)C)CC2)=O)CC(C(C)C)=NO1 c1(C(=O)NCCN(CCCN(C)C)C(C2CC2Br)=O)ccc2ncccc2c1 Cc1cc(C(=O)NC2CCN(Cc3ccc(F)nc3C)C2)cc(C)c1O C1(CCN(C(C(=O)N)c2cn[nH]c2)C)NC(=O)NC1=O.C=C(C)CN(C)C(C)=O c1(C(N2CCC(CN(C)C(C3CCC(O)CC3)=O)C2)=O)ccc2nonc2c1 C(CC(=O)N(CC)OC)C1CCCN(C(=O)NC2(C#C)COC2)CC1 C(C(CC(=O)N1CC=C(CNC(=O)Cc2cc[nH]n2)CC1)C(F)(F)F)N(C)C c1(CC)ccsc1C(=O)NCC1CCC(C(=O)NCCc2ncc[nH]2)C1 C#CC1CC2CCC1N(C(C1CC=CCN1C(=O)CC1COCC1O)=O)C2 Cc1c(-c2cn(CCN(C(=O)CSc3cccc(Br)c3)C)nn2)cccc1Cl C(c1ccc([N+](=O)[O-])cc1)=C(C(=O)OCC(NOCOC)=O)C C(C(=O)NCC1(O)CCN(C(=O)CC2CC=CC2)C1)(C(C)C)OCC c1(C(=O)NC2CN(C(C(C)O)=O)CC2(C)C)cccc2c1C1CCC2CC1 C(C)(CC(C)(C)C)C1C(C)C1.C1CCC(=O)NCC2(O)CC(C2)C(=O)N1 C1(NC(C(C)SCCCC)=O)CN(C(=O)Cc2ncc(C)[nH]2)C(C)(C)C1 C=CCC(C(=O)NC1CCCC1NC(c1[nH]c(O)nc1C)=O)OC c1(N(C2CC3CNC2C3)C(C(C)S)=O)c(C(F)(F)F)cc(Cl)cc1[N+](=O)[O-] C1(C(=O)NC(C(N2C(C)(CCO)CC2)=O)C2CC2)CC2(CCO1)CC2 c1(OC)ccc(C(=O)NC(C)CCCNC(=O)C(F)OC(F)(F)F)nc1 C1(Cn2cc(C3(C)CCCC3)nn2)CCCCCN1C(C12CC(C(F)F)(C1)C2)=O c1(CC)sc(=N)[nH]c1C(=O)NCC1CCCCN1C(c1c(OC)noc1CC)=O c1(C(N(CCCNC(C(C)(C)OC(C)C)=O)C2CC2)=O)cnc2occc2c1 C1(C(=O)NCC(C2CCC2)NC(CC(C)(C)C#N)=O)CCCC2(CCC2)C1 c1(C(C(=O)NCC)N(CC(C)C)Cc2ccc(CSCC)cc2)ccc(Br)cc1 c1(C(C)C)ncc(C(=O)NCC2CCCC2NC(c2coc(Cl)c2)=O)s1 c1(C(=O)NCC(CNC(c2cnc(OC)nc2C)=O)F)cccc2cnsc12 C(=O)(C(O)CC(N)=O)N1CCC(CNC(c2c(C)cc(C)s2)=O)C1 c1(C(=O)NCCOCCN(C(C(C)OCCC(C)C)=O)C)cccc2ccoc12 C1(O)(CC(=O)NCCCNC(c2ccc(C(C)C)s2)=O)CCOCC1 CC(CC(=O)N(C)C)NC(=O)COC1CN(C(c2nnsc2N)=O)C1 c1(CC#N)cccc(C(=O)NCC2COCC2NC(c2ccoc2Br)=O)n1 N1(C(C(C)Cc2cnn(C)c2)=O)CCC(C)(NC(=O)CCc2ccc(O)cc2)C1 C1(c2c(C(=O)OC)nco2)CCN(C(=O)NC2COC(c3ccccc3)C2)CC1 c1(C(=O)NC2(C)CC(NC(=O)CC3(CO)CC3)C2)cc(F)ncc1Br C(CCC(C)(C)C(=O)N1CC(F)(F)C1C1CC1)NC(C1CC=C(C)C1)=O C1(N(C(=O)Cn2ncnn2)CCC)CCN(C(=O)CSC(F)F)CC1 C(=O)(C1=CC2(CCOC2)C1)N1CC(NC(c2ncc(C)c(C)c2)=O)C(C)C1 c1(OC(CC)=O)cc(Nc2cccnc2C(F)(F)F)cc(I)c1 c1(OC)cc(CNC(=O)C=C(C2CC2)C2CC2)ncn1.C12C(CC1O)NC2 c1(CC(=O)NC(C(C)NC(c2c(C)nsc2)=O)C)ccc2c(c1)CCCS2(=O)=O c1(N(C2C(C#N)CNC2)C(c2cc(Cl)cc(Cl)c2)=O)ncnc2c(Br)csc12 Cn1cnc2cc(C(N3CCC(N(c4ncc(Br)cn4)CCO)CC3)=O)ccc2c1=O CCC(CC(F)(F)F)C(=O)N(C(C)CN(C)C(c1c(C)ccc2nn[nH]c12)=O)C NS(=O)(=O)c1ccc(C(=O)NC2CCCC(NC(=O)CC34CC(CCO3)C4)C2)s1 Cn1ncc(C(=O)NCCC2CCCCN2C(=O)CCOc2cccnc2)c1Cl c1(C(=O)OC)c(-c2ccco2)csc1NC(=O)NCC1(c2ccccc2O)CC1 c1(C(=O)NC(C(C)NC(c2cnc(O)c(Cl)c2)=O)CO)cc2cn[nH]c2cn1 c1(N(C(C)C)C(=O)NCc2ccnc(C(F)(F)F)n2)nc2ccccc2[nH]1 c1(C(=O)NCc2c(CC)cccn2)cc(OC)nc(Cl)c1.C12CC(C1)C(=O)NC2 c1(C(N2CCCC(n3cc(C(C)OCC)nn3)C2)=O)cccc2occ(Br)c12 CC1(C)C(NC(=O)CN2CCC(CO)CC2)CCN1C(=O)CCn1cncn1 Cc1ccc([N+](=O)[O-])cc1NC(=O)CN1C(=O)CCC1C c1(C(N2C(C3(O)CN(C(C4CC4F)=O)C3)CCC2)=O)ccc(C2(F)COC2)cc1 c1(C(N2C3(CNC(CC4(C)CC4(F)Cl)=O)CC(C2)C3)=O)ccc(N)c(C2CC2)c1 C1(CNC(C2(C)CC=CCO2)=O)CN(C(=O)COCC2CCC2)CC1(F)F c1(CC)ccc(F)c(C(N2CCOC(CNC(=O)CC3SC(=N)NC3=O)C2)=O)c1 C(=O)(CS(=O)(=O)c1ccccc1F)N1CC(C(C)NC(=O)CCc2cccnc2)C1 c1(C(N2CCCN(C(CC(C=C)CC)=O)C(CO)C2)=O)nc2nccc(C)n2n1 c1(C(=O)NCC2(F)CC(NC(C(C#C)(C)C)=O)C2)ccc2c(c1)COC2 C1(CN(C)C(C2CC3(CCC3)C2)=O)CCCCN1C(=O)CCSc1ccccn1 Cc1ccc(C(=O)NCC2CCCN(C(=O)Cc3nnc(S)n3C)C2)c(Cl)c1Cl Cc1cccc(CC(=O)NC(C)CCCNC(C2CC2CCOC)=O)c1 N1(C(CCC)=O)CCCC(C)C1CNC(c1cc(O)ccc1OC(F)F)=O C12(CNC(c3nccc(OC)c3N)=O)CCC(CC1)N(C(C1(C)CC1(F)Cl)=O)C2 n1(-c2ccc(OCC)cc2F)cnc2ncc(C(=O)N(CCCO)C(C)C)cc12 CC(C)S(=O)(=O)CC(=O)NC(C)C(CO)NC(C1CCN(C)CC1)=O Cn1[nH]nnc1=NCCN1CCN(C(=O)C=Cc2cc(Cl)cc(Cl)c2)CC1 c1(C(=O)NC(CNC(c2cc(C(C)O)sc2)=O)(C)C2CC2)ncn2ccccc12 C(CCS(N)(=O)=O)c1n(CC(C)C(=O)NC(C)(C(=O)O)c2cccnc2)ccn1 N(C(=NCCC1CCCC1)NCC1CCCN1C)CC(C)C c1(-c2nc(C)on2)cccc(C(=O)NCC=C2CCN(C)C2)c1 c1(NC(=O)NC2C(CC)CCCC2)cc(C(=O)NC)ccc1C C1(CN(C)C(C2(n3cccn3)CCCC2)=O)CCN(C(=O)CC2CCOC2)CC1 C1(C(=O)Nc2c(C)ccnc2)CN(C(c2ncccc2Cl)=O)CCN1C N(C(=NCC1CC1)NC1CC1(C1CCOCC1)C(=O)N(C)C)C1CC(COC)C1 C1(NC(C2(C(C)NC(c3cccc(C)c3C)=O)CC2)=O)CCc2ncnn2C1 CC1CCC(CNC(c2cccc(-c3nc(O)n[nH]3)c2)=O)CN1C(=O)CNC=O CCCC(CCC)C(=O)N1CCCC(COC)(NC(c2cscc2CC)=O)C1 C1(NC(C(Br)=C(C)C)=O)CC(F)CN(C(c2cc(C(F)F)n(C)n2)=O)C1 C1(C(=O)NC(C#C)(C)C)(NC(c2occc2CC)=O)CCCC1C n1(CCOCC)ncc(NC(c2cccc(CNc3cnc(C)[nH]3)c2)=O)c1C Cn1cc(CC(=O)NC2CN(C(=O)CC3CCCC(=O)N3)C2)c2ccccc12 C1(CN(C(c2cc(COC)[nH]n2)=O)CC)CCN(C(c2ccccn2)=O)C1 N1(C(c2c(C)nc(CO)nc2)=O)CCC(NC(=O)C(C)C(C)C)C2(CCC2)C1 CCC(CC)C(F)C(=O)N1CC=CC1C(=O)NC1CC12CCCCCC2 C(=O)(C1=C(C#N)CCC1)N1C(C)CCC(C(=O)NCCN2CC(C)(O)C2)C1 C(=O)(CCCCC(=O)N1CC(CO)(NC(=O)C(C)(F)F)C1)OC CC1=CCC(C(C)CC(=O)NC2COCCC2NC(c2sccc2CO)=O)CC1 CC1CCCCC1(CNC(=O)Cc1ccccc1)NC(=O)COC1CCCOC1 Cc1cc(Cl)cc(NC(=O)CCC2CCCN2Cc2ccc(I)cc2)c1I C1(CNC(COc2cn(C)nc2)=O)CCCN(C(=O)CC(F)F)C1 N1(CC)CC(C(N2CCN(C(c3ccccc3)=O)C(C(F)F)C2)=O)CCC1=O CC(C)CC(C(=O)NCCC(C)c1cn[nH]c1)ONC(=O)C1CC(F)C1 N1(C(Cc2nc(C)cc(C)n2)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C2CCC12 CC1(C)CC(C)(CNC(=O)CC2CC2(Cl)Cl)CN1C(C1CC2(CCC2)C1)=O c1(C(C)OC)nc(C(=O)N(C)Cc2cn(CC3C(C)C3(F)F)nn2)co1 Cc1nncc(C(=O)NC2C=CCN(C(=O)CCCF)C2)c1C C1(CNC(CCn2cc(-c3c(C)ncs3)nn2)=O)(CO)CCCCC1 c1(C(C)C)nc(C(=O)NCCC2(O)CN(c3nnnn3C)C2)cs1 Cc1cc(C(=O)NC2(C)CCCN(C(c3ccc(Cl)c(CO)c3)=O)C2)cc(C)c1 c1(C(C(C)O)NC(=O)NCS(=O)(=O)c2ccccc2)nnc2ccccn12 C=CC(CCC)CC(=O)NC1COCC1NC(c1cnc2ccnn2c1)=O CC1CCN(C(=O)COCCN(C)C)CC1NC(c1ccnnc1O)=O C(=O)(CCC(C)(C)CNC(c1csnn1)=O)OCC C1(NC(CC2(C)CCCO2)=O)CC12CCN(C(=O)COCCCF)C2 C1(CNC(c2cc(CC)[nH]n2)=O)(NC(c2cc(C(N)=O)c[nH]2)=O)CCC(F)(F)CC1 O=C(Cc1ccc(I)cc1)NNC(=O)c1ccnc(C2CCCC2)n1 c1(C(=O)NCC2CC(NC(CSSC)=O)C2)cn2cccnc2n1 c1(C(C(=O)NC(C)(C)CC)N(C(C#C)COC)C)cn2cc(Br)ccc2n1 c1(OC)cc(C(=O)NC2CN(C(=O)CCCn3cccn3)C2)cc2cccnc12 C1(CCOC)CN(C(=O)CC2=CCCC2)CCN1C(c1ncn(C)c1C)=O C(CC(C(C)C)NC(=O)Cn1cc(Br)c(C)n1)N(C(CCC)=O)C c1(C(C(=O)NCC(C)C)N(C2CC2)CC2CCOC2)ncc(Cl)cc1Br CCC(F)(F)CC(=O)NCC1(C)CCCN(C(=O)CCN2CCC(F)C2)C1 N1(C(=O)OC(C)(C)C)CCC(NC(c2ccnn2Cc2ccccc2)=O)C2CC12 C1(C(=O)NCC2(CNC(c3cnc(O)o3)=O)CC2(F)F)CCCC(CF)C1 C1(C2CCN(C(c3ccc(Cl)cc3N)=O)CC2)(NC(C2C(C)OCC2)=O)CCC1 N1(C(C2CCN(C(C3CN(C4COC4)C3)=O)C2)=O)CCC12CC(O)C2 O=C1CCCN(C(C23CSCC2C3)=O)CC1.C12OCCC1CONC2=O N1(CCC=CCC)CCC(NC(C2(c3cccs3)CCCC2)=O)C(O)C1 Cc1cc(C(=O)NCCC2(C(=O)NCc3cc(C)n(C)n3)CCCC2)ncc1F C1(C(N(C(C)CO)CC)=O)CC2C=CC1N(C(c1ccn(C)c1C)=O)C2 C1(NC(c2ccc(C)n2C)=O)CC2CCC1N2C(=O)CCC1CC(C)(C)CO1 Cc1ccc(Br)c(F)c1C(N1CCC(F)(F)C(NCc2ccc(F)c(F)c2)C1)=O n1(CC(=O)O)cc(CN(C(=O)CCO)O)nn1.C(COCCOCCNC=O)OC.C(C)OC CC#Cc1ccc(C(C(=O)NCCCF)N(C2CC2)C(C)C)cc1 N1(C(CCC(=O)NCCC)=O)CCC(NC(c2ncc(C)cc2F)=O)C(O)C1 c1(OC)ccc(C2CC2C(=O)NN2CCC(Cc3[nH]ncc3C#N)C2)cc1 CC#CCCCCN=c1ccnc(NCc2ccc(-n3cc(Br)cn3)cc2)[nH]1 CC1(C)C=C(C(=O)NCCCNC(=O)CCCSc2ccc(Cl)cc2)C1 CC(C)C(=O)C(=O)NC(C1CCCN1C(C1CC2CCC2C1)=O)C N1(C(C(CC)=O)=O)CC2CN(Cc3cc(Cl)cc(Cl)c3O)CC2C1 CC1(C)C(=O)NC(NC(N2CCCCC2)=O)C(=O)N1C1CC1 C1(CNC(CC2(OC)CCCCC2)=O)CCC12CN(C(=O)CC1CC=CC1)C2 c1(C(=O)NCC(C)(C)NC(c2ccc(CC)[nH]2)=O)ccc(S(=O)(=O)CCO)cc1 c1(CN2C(CCN(CC(=C)Br)C)CCCC2)ccc2nc(O)[nH]c2c1 N1(C(COCCC=C)=O)CCN(C(c2cc(Cl)no2)=O)CC12CCC2 Cc1ccc(F)c(NC(N2CC3CCC3(CNC(c3cncc(F)c3)=O)C2)=O)c1 C1(CN(C(=O)CCN2CCOC2=O)C)CCCN(C(c2ccsc2)=O)C1 c1(C(=O)NC2CCC(NC(CCC(C)NC(N)=O)=O)C2)cc(N)cc(F)c1 N1(C(C(C=CC)O)=O)CCC(O)C(NC(c2cnnc(C)c2)=O)C1 CC1CCCN(C(=O)C(C)n2ccnc2)C1CNC(c1cc(O)ccc1Cl)=O C1(CNC(CCC=C)=O)CN(C(=O)Cc2cccnc2)CCC1(C)C C(=O)(C(C)C1=CCCC1)NCC(C(C)C)NC(c1c(OC)c(Cl)ccc1)=O C12CC(CO1)C(=O)N2.C1(NC(c2nocc2Cl)=O)CCN(CCF)C1 C1(CN(C(=O)CCCN(C)C)C)CN(C(C2C(C)(C)C2(F)F)=O)CCO1 CC(CC(C)(C)C)C(=O)NC1(CO)CCCN(C(=O)CC2CCCC(C)(C)C2)C1 c1(C(=O)NCC(CNC(c2[nH]ccc2C)=O)OC)ccc(OC(F)(F)F)cc1 C1(C2(O)CN(C(=O)C=C(C)C)C2)(CNC(c2cc(OC)c(OC)nc2)=O)CC1 CC1(C)CN(C(c2cnc(S)[nH]2)=O)CC(CNC(c2cc[n+]([O-])cc2)=O)O1 c1(NC(C(=O)NCC(N2CC(C)=C(C)CC2)=O)=O)cc(C)c(F)c(S(C)(=O)=O)c1 c1(C(=O)OC)cc(=NC(CCN(C(=O)C(O)C(C)(C)C)C)C(C)C)[nH]c(Cl)n1 CC(C(=O)N1CCN(C(c2sccc2-n2ccnn2)=O)CC1CCO)C(C)(F)F Cc1cc(=NCC(c2cn(C)cn2)NC(C2(C(=O)N(C)C)CC2)=O)[nH]cn1 CC1(C)CN(C(=O)CC2(O)CCCOC2)CC1CN c1(CC)cc(Br)ccc1C(N1CCCCC1C(N1CCN(C2CC2)CC1)=O)=O c1(C(=O)NCCC2(C)CCN(C(C(CC)(C)O)=O)C2)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)NCCCC(C)NC(c2cccc(F)c2Cl)=O)c2c(nn1C)CCSC2 N1(C(C=CCC)=O)CCC(NC(=O)CN(C(=O)CC(O)CC)CCCCC)CC1 C1(NC(C(C)NC(=O)OCC)=O)CCCCC1NC(c1cnc[nH]1)=O C(=O)(CCCC(C)(C)N(C)C)NC(C)Cn1cc(-c2ccc(Cl)nc2)nn1 C1(CNC(C2CC3(CCC3)C2)=O)CN(C(c2csc(-c3nc[nH]n3)n2)=O)CCO1 C(N=c1[nH]c(=NC(C)c2cn[nH]c2)[nH]c2ccc(Cl)cc12)c1c(C)ccc(Br)c1 c1(C(N2C(C(C)NC(=O)CNC=O)CCC2)=O)cccc2c1ccn2C N1(C(C2CC(OC)C2)=O)CCC2(CC(NC(C3CC(OC)C3)=O)CO2)C1 CN1CC(NC(=O)C(C)(C)CN(C)C(c2ccc3c(c2)CC3)=O)CCC1=O C1(C(=O)NCC(CO)NC(C(CC2CCC2)OC)=O)CCCCN1N=O c1(OC)ccc(C(=O)NC2CC2C2CN(C(c3cccnn3)=O)C2)c(F)n1 CCC(O)C(C)C(=O)N(C)CC1CCCN1C(=O)CNc1ccccn1 c1(NC(C2CC(C(F)F)(OC)C2)=O)cccc(CNC(=O)CNS(=O)(=O)N(C)C)c1 C1(N(C(CSCC#C)=O)C)CCCC(N(C)C(c2sc(CC)nc2C)=O)C1 N1(C(c2ccnc(OC)n2)=O)CCCC(F)(CNC(C2CC2C(=O)NC)=O)CC1 C1(NC(C2C(CNC(C(C)SC)=O)C2(C)C)=O)CCC2CC1C2(C)C c1(NC(N2CC(C)(C(=O)NC(C)CC3CCOC3)C2)=O)ccc2sccc2c1 C1(NC(C2C(C=C)OCC2)=O)CC2CCC(C1)N2C(c1ns[nH]c1=O)=O c1(CC)cc(C(=O)NCC2CC(OC)CN2C(=O)CC(C)n2cccn2)cc(Cl)n1 CC1CCCc2c(C(=O)N(C(C)CCNC(c3sc(F)cc3Cl)=O)C)cnn21 C(=O)(CS(F)(F)(F)(F)F)N(C1CCCN(C(=O)CCN(C)CCO)C1)C O=C1NCCC2=C1C(c1csc(-c3ccco3)n1)NC(=S)N2Cc1ccco1 Cn1cc(Br)c(CC(=O)NCC(C)(C)NC(=O)CCN2CCCS2(=O)=O)n1 c1(OC)cc(F)ccc1C(=O)NCC1(CNC(=O)Cn2nc(C)nc2C)CC1 c1(C(N(C2CCCC2)CCNC(CCCOC)=O)=O)cc2sc(Cl)cc2[nH]1 Cc1c[nH]c2ncc(C(=O)NC(C)C(C)NC(=O)C=Cc3ccco3)cc12 C1(CN(C(c2ncccc2O)=O)CC)CCN(C(=O)Cc2ncoc2C)CC1 c1(C(=O)NC(C2(O)CN(C(=O)CNS(C)(=O)=O)C2)C)cc2ccsc2c(O)n1 c1(C(=O)NC(CN(C(c2c(OC)nsc2OC)=O)C)C)cccc(N)c1N C12(C(=O)NCC3(C)CCCOC3)CC(CO1)N(C(=O)CN1CCCNC1=O)C2 N1(C(Cc2ncc(C)[nH]2)=O)CCC(N(C(=O)Cc2cnccn2)C)C(C)C1 C1(NC(c2nc(COC)oc2)=O)CCN(C(C2(C(F)F)CCC2)=O)CC1 CCC(C)(C)C(=O)NC(C1CN(C(c2c(COC)ocn2)=O)C1)C CC1CCCN(C(=O)CCC2CC(NC(C3CN(C(N)=O)C3)=O)C2)C1CO c1(C(N(CC(CNC(C(CC=C)NC(C)=O)=O)C)C)=O)cnc2scc(C)n12 c1(C(N2C3CC(NC(Cc4cncc(C)c4)=O)(C3)C2)=O)ccc(Cl)cc1C C1(CC(=O)NC(CCC)C2CC2)CCCN(C(C2(C3(O)CCC3)CC2)=O)CC1 C1(NC(C=CSC)=O)CC12CCN(C(c1cc(NS(C)(=O)=O)cc(F)c1)=O)CC2 c1(C(N(CCCNC(=O)CN2CCCCC2=O)CC)=O)cccc(C#N)c1 CC(C)CCCCC(=O)NCC(C(C)(C)C)NC(C1(O)CC(C)(C)C1)=O C(CC(O)C(=O)NCCC(C)N(C(=O)C(=O)NCc1ccccc1)C)SC CCC(CN(C)C)CC(=O)NCc1ncc(C(=O)NC2CCC2O)cn1 c1(CC)ccc(F)c(C(=O)NC2CC(C)(NC(=O)Cn3nc(C)cc3C)C2)c1 N1(C(CCSC)=O)CC2(CCCCN2C(c2nccn3cc(C)nc23)=O)C1 Cc1sc(C(=O)NC2CC(F)(F)CC2NC(=O)CC(C)F)cc1[N+](=O)[O-] N1(C(CC2N(C(c3n(C)cnc3)=O)CC2)=O)CCCC(O)C1 c1(NC(C)=O)cccc(C(N2CC3CC3(CNC(=O)CC3CCCO3)C2)=O)c1C CC(C(=O)NCCC1CCCCN1C(=O)CCCc1cncs1)S(C)(=O)=O C1(C(N)=O)CN(C(=O)Nc2cc(F)ccc2N(C)C)CCN1CCOCCO CC(CCCCO)NC(c1coc(CNC(C2CCC2C(C)(C)C)=O)n1)=O c1(C(=O)NC2CCCC2CNC(C2CCO2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C(C(CNC(c1cscn1)=O)S(C)(=O)=O)NC(CC1CN(C)C1)=O N1(C(C(C(=O)OCC)C(C)C)=O)CCC2(CC1)CCN(C(=O)CCCC(C)CC)C2 C1(C)(C(N(CC)CC)=O)CC12CCN(CC(F)(F)F)CC2.C12CCCN(C1)C2=O N1(C(c2c(OC)c(F)ccc2)=O)CCC2(CCCN2C(c2cccc(=O)o2)=O)C1 c1(COC)cc(CC(=O)NCC2CCC(NC(=O)CCc3cnc(O)[nH]3)C2)no1 N1(C(C2(C)CCN(C(=O)Nc3c(C)ccc(C)c3)CC2)=O)CC2CCCCC2C1 c1(NC(CC2N(C(C3CCC(CC)O3)=O)CCC2)=O)cnc2ccccc2c1 c1(CC(=O)NC(CN(C(c2cc(CO)[nH]n2)=O)CC)C)cn(C)nn1 CCC(CO)(C(=O)NC1CCC(N(C(=O)C(O)C(C)(C)C)C)CC1)OC Cc1cnc(N2CCOC(C(=O)NCCc3cc(O)no3)C2)nc1C CC1(F)CCCN(C(C2CC(O)CN2C(=O)COC2CCCOC2)=O)C1 C12(C(=O)OC)CCC(C(=O)OCCCCn3cc(C(C)OC)nn3)(CC1)O2 C1(NC(CCC)=O)CCCCC12CN(S(=O)(=O)c1ccc(F)c(F)c1)CCO2 CC(C)CC(O)C(=O)NC1(CNC(c2nn(C)cc2C(F)(F)F)=O)CCC1 c1(-c2n(C)ncc2)cnc(Cl)c(C(=O)NCC2(O)COC2)c1 Cc1[nH]nc2cc(C(=O)NC3CN(C(c4ccc(N)c(F)n4)=O)CC3O)ccc12 N1(C(C2CCC(=O)O2)=O)CCCCC(C(N2CCCCC(N(C)C)C2)=O)C1 C(=O)(CCC(C)S(C)(=O)=O)NCC1(CNC(C(CCC)CC)=O)CCCC1 c1(OCC)ccc(N)c(C(=O)NCCN(C(c2ncccc2F)=O)CC)c1 N1(C(CSCC)=O)CCC2(CCN(C(=O)CSc3c(C)noc3C)CC2)C(C)C1 N1(C(c2c(OCCC)cccn2)=O)CC(C2(NC(c3nc(C)sc3C)=O)CC2)C1 C12(CNC(=O)CN3CC(=O)NC3=O)CCCC1N(C(=O)Cn1nccn1)CCC2 c1(OCC(=O)NCC2CCC2NC(=O)CN2C(=O)CNC2=O)cccc(O)c1 N1(C(C2C(CC(C)(C)C)C2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC12CCCC2 C1(NC(c2nc(C(N)=O)sc2)=O)CCN(C(=O)CCn2cccn2)CCC1(F)F C(=O)(C(F)C(F)(F)C(F)(F)F)N(CC(C)O)CCNC(C1(F)CCCCCC1)=O Cc1cc(C(=O)NCC(C)(C2CC2)NC(C2CCOC2C)=O)cc(C)c1 CN=c1cc(C(N2CC(CNC(=O)CCc3ccsc3)C(C)(C)C2)=O)cc[nH]1 CN1CCN(c2ncccc2CC2CCCN(C(c3cn(C)cn3)=O)C2)CC1 O=C(C#Cc1ccc(Cl)cc1)N1CCc2cc(C(=O)NC34CC(C3)C4)ccc2C1 N1(CC(=O)N(C(C)C(=O)N(C)Cc2ncco2)CCC)C(=O)CCC1=O c1(OC)cccc(I)c1NC(C1CC(Nc2ncc(-c3ccccc3)cn2)C1)=O c1(C(=O)NCCC2CCN(C(=O)C=C3CCCC3)CC2)cccn2c(O)nnc12 C1(CNC(C(C)NC(=O)C(n2cc(CCCCO)nn2)C)=O)CCCCN1C CC1c2ccccc2OC1C(=O)NCC1CN(C(C2CC(n3ccnn3)C2)=O)C1 C(CN=c1ccnc(NCC(N2CCCC2)=O)[nH]1)(c1ccc(OC)cc1)OC N#Cc1cc(Cl)c(C(=O)NCC2(NC(=O)Cc3nc[nH]n3)CCOCC2)s1 c1(C(c2nc(NC(N3CC(c4ncccn4)(C)C3)=O)sc2)=O)ccc(F)cc1 c1(C(N2CC(F)(CNC(C(CC)NC(C)=O)=O)C2)=O)c(C)nn2c1CCCC2C c1(OC(C)C(=O)N(CCCN(C(=O)C(C)(C)C(N)=O)C)C)ccc2c(c1)CCC2 N1(c2cc(N3CCCC(C(=O)OC)C3)ncn2)CCCc2[nH]ccc2C1 Cc1cccc(C(=O)C(=O)NCC(C)NC(c2cn(C3CCC3)nn2)=O)c1 C1(NC2(CCNC(c3ccc(-n4cccn4)nc3)=O)CC2)CCS(=O)(=O)C1 C1(C(N2CCC(CNC(C3CCC(C(=O)OC)CC3)=O)C2)=O)CCCCN1N=O C(=O)(C(C)CC(C)(C)C)N(C(C(=O)NCC1(C#C)CCOCC1)C1CC1)C C1(C)(C(=O)NC2CC(NC(C(CCSC)O)=O)C2)COC(C)(C)CO1 c1(CCC)ccc(CC(=O)NC2(CNC(=O)COC(C)C)COC2)cc1 C12(C(=O)NCCSCC(=O)OCC)CC1COC2(C)C CC1CCN(CC(=O)N(CCN=[N+]=[N-])CCCC2(O)CCCCC2)CC1 C1(C(=O)N(C)CC2CN(C(c3cccc(C(C)C)n3)=O)C2)C2CC3C(C2=O)C13 N1(C(CCCCC#C)=O)CCC(C(=O)NC2CC(C3CCC3)C2)CC1(C)C c1(C(=O)NC(C2CN(C(C3CC(SC)C3)=O)C2)C)cc(Cl)c(F)cc1Cl N1(C(c2c(C)cccn2)=O)CC(NC(=O)C(C)c2ccon2)CC(C)C1 CC1(NC(C23CCCC2C3(F)F)=O)CCN(C(c2cocn2)=O)CC1 Cc1c(Cl)ccc(C(=O)NC2(C3CN(C(=O)Cc4c[nH]ccc4=O)C3)CC2)c1O C1(OC)CC(NC(=O)CCCN2C(=O)CCC2=O)CN(C(C2CNC(=O)C2)=O)C1 CCCCCC(C)(CC)C(=O)N1CCC(=O)N(C)CC1.c1cn(CC(O)CO)nn1 c1(C(N2CC(CNC(C=CC(C)(C)C)=O)C3C2C3)=O)ccc(F)c2ccsc12 C1(C(=O)NCCC(C)(C)NC(c2coc(C3CC3)n2)=O)CCS(=O)CC1 c1(C(=O)N(C)CCN(C(=O)CC2CCC(C)O2)C)c[nH]nc1C1(CC(C)C)CC1 N1(C(c2cnc(C(F)(F)F)s2)=O)CCN(C(c2coc(Cl)n2)=O)C(C(F)F)C1 C1(NC(c2c(C)noc2)=O)C=CCN(C(=O)COCC(C)(C)C)C1 C1(C(=O)OCC)CCN(C2CCC(N)C2)C1 CCC(COC)C(=O)NCC(C1CCCC1)NC(C1(N(CC)CC)CCCC1)=O C(=O)(C(C)(C)c1cnco1)NC(C)COC(F)F n1(CC=C)cc(C(=O)N(C2CCC(NC(=O)C=CBr)C2)C)nn1 Cn1ncc(Cl)c1CCNS(=O)(=O)CC1CCCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2(C#N)CCN(C(c3cnccc3Cl)=O)C2)cc2cccnn2c1 N1(C(c2c(SC)ccs2)=O)CC(NC(C2(CCF)CCOCC2)=O)CC1(C)C c1(NC(c2c(NC3CC(=C)C3)cccn2)=O)nc(C)ncc1Br CCC(C)(C)C(O)C(=O)N1CCC(C)N(C(c2occ3c2CCOC3)=O)CC1 N1(C(c2cncc(C#C)c2)=O)CC(C)CN(C(=O)CN(C)CCO)CC1C CC1COCCCN1C(=O)C(Cn1cccn1)NC(c1ccn2ccccc12)=O CCC1=C(C(=O)NC2CC3CC2CN(C(C2CCCCC(=O)N2)=O)C3)CCCO1 C1(O)(CC(=O)N(C)Cc2ccccc2)CCN(C(C2CCCCC2N)=O)CC1 C1(CNC(C2C3CC4C(C3)C24)=O)CC2(CCN(C(c3ccc(Cl)cn3)=O)C2)CO1 N1(C(CC=C)=O)CC(F)(F)CC1CCNC(=O)COc1c(C)nn(C)c1C C1(NC(=O)Cc2nc(C3CC3)n[nH]2)CCSC12CN(C(c1ccc(O)cc1)=O)C2 N1(CC)CC(NC(C2(C)CCN2C(C2(OC)CCCCC2)=O)=O)CC1=O C1(C(=O)NC(c2cn(C)nn2)C(=O)NCc2nnc(C)o2)COCCC1C C1(C(=O)NC2C(NC(c3c[nH]nc3C(F)(F)F)=O)C2)C2CCC(F)C12 N1(C(c2nccc(CC)c2)=O)CCC2C(CCN2Cc2cccc(O)n2)C1 Cc1ccc(C(=O)NCC2(F)CCCN(C(c3cnsc3)=O)C2)c(C)c1 C(C(=O)NC(Cc1ccoc1)C(=O)Nc1cccc(C(C)F)c1)(C(C)C)OCC c1(OC2CN(C3CCC3)C2)ccnc(NCC(=O)OC)n1 c1(C(=O)NCC2N(C(C(CC)OC)=O)CCCC2)ccc2c(n1)CCCC2 N(C(=NCc1ccccc1F)N(C)Cc1cccn1C(F)F)C(C)C Cc1cnc(C(=O)NC2CC(C3=CCOC3)S2)cc1C C(C(C)C(=O)N1CCCC1CN(C)C(C1C=CCS1)=O)OC(C)=O CCCCS(=O)(=O)CC(=O)NC1CCN(C(=O)C(F)(F)CCn2cccn2)C(C)C1 C(=O)(C1=CCCN(C(=O)C(O)C2CC2)C1)NC(c1c(C)nccn1)C N1(C(C2N(C)CCOC2)=O)CCN(C(c2ccc(N)c(F)n2)=O)C(CC2CC2)C1 C1(C)(C(N(C)CC2CCCN(C(=O)C(N)=O)C2)=O)CCN(S(N)(=O)=O)CC1 c1(C(N2C(C)CC(NC(c3cc(CC)no3)=O)C2)=O)ccc2nn[nH]c2c1 c1(C(=O)NC2CC2NC(N2CCCC2)=O)cc(O)ccc1F.O=C1CCCCN1 n1(CC)cc(CNC2(C)CN(C3CC3)C2)cn1 N1(CC)CCCCC1C(=O)NC1CCCCC1CNC(C1CCCCNC1=O)=O c1(SCC(=O)NC(C(C)NC(c2c(CC)cno2)=O)C)ccc(Cl)cc1 c1(C(C)NC(C2(NC(=O)Cc3nc(=N)[nH][nH]3)CSC2)=O)scnc1C CCC(CC)C(=O)NCCOCCNC(=O)C(C)(C)n1cc(Br)cn1 c1(C(=O)NC23C(NC(C4C(C=C)CC4)=O)CC(CC2)C3)ccc2cnccc2c1 C1(NC(CCNC(=O)C=CCl)=O)CC(NC(c2cc(Cl)ns2)=O)C12CCC2 CC1(C)CCCC1(C)NC(C1CCC1CNC(=O)CNC(=O)OC)=O CCCC(C)C(C(=O)NCC)N(C1CCN(C2CC2)C1)CC(C)(C)C c1(C(=O)O)ccc(-c2ccc(C(F)(F)F)nc2Cl)n2nccc12 C1(CC(N2C(C(=O)NCCC3(OC)CCC3)CC2)=O)CCC(=O)C1 C(=O)(C1CCCc2sccc21)N1C(CC)(CC)CC(NC(C2CS(=O)(=O)C2)=O)C1 c1(SC)ccc(CNC2CC(CNC(C3CCC3)=O)C2)cc1 C1(C2CCN(C(C3CCN(C(N)=O)CC3)=O)C2)(NC(CC2CCN(C)C2)=O)CC1 c1(C(=O)NCCN(C(=O)Cc2ncc(Cl)s2)C2CC2)cnc2n1CCS2 c1(CC(C(=O)OCc2cnoc2C2CCC2)O)cc(Cl)ccc1Cl C(=O)(C(CC)CCOC)Nc1c(OCC)cccc1.C1(=O)C(C)N2CC(C2)CN1 c1(C(=O)NCC2N(C(CC(CCC)(C)O)=O)CCC2C)nc2nc(C)ccn2n1 c1(-c2cnc(C3CN(C(CN(C4CCOCC4)C)=O)C3)o2)cccc(C#N)c1 N1(C(CN(C)CC)=O)CCOCC(NC(c2cnoc2C2CC2)=O)C1 c1(N2CCC(C)OCC2)nc(=N)[nH]c(=NCc2cscc2C(F)(F)F)[nH]1 N1(C(C(C)(C)c2ccns2)=O)CCC(NC(c2ccc(F)c(N)c2)=O)C(CO)C1 N1(C(c2ccc3c(c2)N(C(C)=O)CCC3)=O)CCc2nc(C#N)ccc2C1 NS(=O)(=O)c1cccc(NCCCNC(N2CCC3CC23C(F)(F)F)=O)c1 CC1(C)CN(C(c2coc(O)n2)=O)C(CNC(c2nccnc2C(N)=O)=O)CO1 C(C)(CCC(=O)NCCC1(CNC(=O)C(C)COCC)CC1)OC C=CC1(C(=O)NCCCC2CC2C)CCN(C(=O)Cn2nccn2)C1 c1(C(C)C)ccc2c(c1)CCN(CCSC1CCCOC1)C2 c1(C(=O)NCCC#C)cnc(-c2ccccc2)[nH]1 CC1C(NC(=O)Cc2cccc(Cl)c2F)CCCN1C(=O)CC(C)(F)F CCC(CC(=O)NCc1c[nH]nc1C(=O)NCc1ncn(C2CC2)n1)C(F)F N1(C(=O)CNC(=O)C(c2cc(F)cc(F)c2)(F)F)CC2CCC(C1)N2 N1(C(C2(C=C)CCC2)=O)CC(NC(=O)CCc2ncc(F)cn2)C(O)C1 C1(CC(=O)NCCOCC(F)F)CN(C(=O)CCCC)CCO1 c1(C(=O)Nc2nc(Br)ccc2Br)cnc2c(-c3cccc(O)c3F)cnn2c1 N1(C(C2CC(C(=O)OC)C2)=O)CC(Nc2ncnc(O)c2Br)CC2(CCC2)C1 C(=O)(C1=C(Cl)CCOC1)NCCC1N(C(C2C(C)(C)C2)=O)CCCC1 c1(NC(C2CC(=C)CN2C(C2(C(=O)OC)CCC2)=O)=O)cc(F)ccc1I O=S(=O)(c1ccc2[nH]c(=NCC34CCCC3C4)sc2c1)NC1C2CCCOC12 N1(C(c2c(C)cncc2)=O)CCCC2C1CCCN2C(C1CC(CF)C1)=O n1(CC(=O)NC(CCNC(CC(C)OC)=O)C)c(C)cc2ccccc12 c1(-n2cc(CCNC(c3occc3C3CC3)=O)nn2)cccc(Cl)n1 C(=O)(C(F)C(C)(C)O)NCc1cccc(CNC(c2csc(C)c2C)=O)c1 CCCC(C(=O)NCc1nocc1C(=O)NCCC1CC2CCC1O2)OC CCC(C)C(C(=O)NC1(C(=O)N(C)Cc2noc(C)n2)CCOCC1)N(C)C C1(NC(c2c(NC(CC)=O)cccc2)=O)CCN(C(c2occc2C)=O)CC1O C1(NC(=O)CCC2CCCOC2)CCC(n2cc(C3CCC3)nn2)CC1 Cc1cc(C(=O)NCCN2CCN(C(c3nc(=N)cc[nH]3)=O)CC2)nn1C(C)C C(CC(C)C(=O)NC1(CF)CCN(C(c2cccc(C(N)=O)n2)=O)C1)=CCC C(C(C(=O)N1CC(NC(=O)C(C2CC2)OCC)C1)OC)OC c1(C(=O)NC2(CNC(COCC(c3ccccc3)C)=O)CC2)c[nH]ccc1=N N1(C(CCC(=O)OC)=O)CCC(NC(=O)Cc2cccc(OC)c2Cl)C(O)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(CNC(=O)CC(C)O)CC12CCC2 N1(C(c2n(CC)ncc2Cl)=O)C2CCC1CN(C(C1C3CCC1(C)C3(C)C)=O)C2 CC(C)C(=O)C(=O)N1CCOC(CNC(=O)C(c2cccc(O)c2)C)C1 Cc1n[nH]c(C)c1C(=O)NCC(C)(C)CN(C)C(c1c(Cl)csc1Cl)=O c1(OC(C)C)ccccc1-c1nc(C(O)C2CC2)n(-c2ccnc(Br)c2)n1 N1(C(C(C)C(F)F)=O)CCC(O)C(NC(c2c(NC(N)=O)cccc2F)=O)C1 C(=O)(C1=CCC(C)CC1)N(CCC(C(C)C)NC(=O)Cc1ccoc1)C N1(C(CCCC#C)=O)Cc2cccn2CC(C(=O)NCc2ccc(C#N)cc2)C1 CC(CNC(=O)CCn1cnnn1)C(=O)N(C1CCCC1)C CCC(C)C(C(=O)NCc1ncc(CO)[nH]1)NC(=O)C=Cc1cc(C)no1 Cc1cccc(CC(=O)Nc2ccc(-c3nn[nH]n3)cc2C)c1C Cc1ccnc(O)c1C(N1CCC=C(CNC(C2CS(=O)(=O)C2)=O)C1)=O CC1CC2CN(C(c3cn(CCNC(c4cccnc4)=O)cn3)=O)CC12 c1(C(N2CCC(O)C2)=O)cccc(O)c1O c1(C)cccc(CO)n1.c1(CCCC)ccc(C(=O)NNC)s1 N1(CCNC(c2c(C)cc[nH]2)=O)CCN(c2nnc(C(N)=O)s2)CC1 c1(CNC(COCCC#C)=O)cccnc1CNC(C1C(C#N)C1(C)C)=O CC(F)(C(=O)N1CCCC(N2CCN(C(C3(C#N)CC3)=O)CC2=O)C1)C(F)(F)F c1(CCC(=O)N2CCCNC(=O)C2)csc(C)n1.C=C1CC1C=C c1(C(=O)NC2CN(C(C3C4CCC3CC4)=O)C2)cccc2c1CCC2 N1(C(C2(CC)CC2)=O)CCCCC(NC(C2(C(=O)NC)CC2)=O)C1 c1(OC)cnc(F)cc1C(=O)NC1CCCCC1NC(=O)C(C)=C1CCC1 C1(O)(C(C(=O)NCCOCC(F)(F)F)NC(CC)=O)CCCCC1 C1(C(=O)NCc2cnccc2Cl)CCC2CCC1N2C(=O)C1=C(Cl)CCC1 N1(C(C2CC(CC)C2)=O)CC2(CCN(C(c3cc(C)n(C(C)C)n3)=O)CC2)C1 C(=O)(CCC(=O)NC1CC1)NC1CC(CCNC(CSc2nc(C)sc2)=O)C1 C(=O)(CCC(C)CN(C)COC)N1CCC(C(Cn2cc(CC(C)O)nn2)F)CC1 S(=O)(=O)(C1CCOCC1)N1CC2C(CNC(c3ccnnc3)=O)(C2)C1 C1(C(=O)NCC2(OCC)CN(C(=O)C=C3CCOCC3)C2)CC2C(C1)C2(C)C c1(OC)ncccc1NC(=O)CC1(OC)CN(C(C2CC(C)CO2)=O)C1 C(=O)(C1CCCn2ncnc21)NC1(CCOC)CCN(C(=O)CC(C)SC)C1 CCC(C)(COC)C(=O)Nc1cncc(CNC(=O)CCc2ncnn2C)c1 C1(CNC(CCc2cc(C)no2)=O)CC(NC(=O)C=Cc2cocn2)CCO1 Fc1ccc(-n2nc(C3CCOCC3)nc2-c2ccoc2)cc1Cl C(=O)(C1(C)CCn2c(C)nnc21)NC(CCCNC(C1(CCOC)CC1)=O)C Cc1ccc(O)c(CNC(=O)CCC2CCCCN2C(=O)C(=O)C(C)C)n1 C(C)(CNC(=O)C(C1CCCCC1)c1cccs1)(CO)NC(COCCCC)=O N1(C2Cc3n(-c4cn(C)nc4)ncc3CC2)CCOC2(CCS(=O)(=O)C2)C1 CC1(C(=O)NCC2CCCN2C(=O)C(=O)NCC2CC2)CCC(=O)NC1 N1(C(C(CC(N)=O)NC(C(C(C)C)N=[N+]=[N-])=O)=O)CCC2=C(CCCC2)C1 C1(C)(C(N(C)CC2OCCN(C)C2)=O)CCCN(C(=O)CSC2CCCN2)C1 C1(NC(C2CCCNCC2)=O)CC2(CCC(F)(F)CC2)C1 N#Cc1cc2c(nc1O)CCN(C(=O)NCC1CC1c1ccccc1Br)C2 c1(CC(N2CC(OC)C(NC(=O)CN(C)C(C)C)C2)=O)cnc2ccccc2c1 N1(CCN(C(CSc2c(C)nns2)=O)OCc2ccccc2F)CCCCCC1 CCC(N=c1[nH]c(=NCC2C3CCCCC23)[nH]c2c1CSC2)C1CCOCC1 C1(C(N(CC#CC)C)=O)CCC2(CC2)N1C(c1cn(C)nn1)=O c1(C(=O)NCC(CCOC)NC(c2cnc(C)[nH]c2=N)=O)onc2c1CCCC2 C1(CNC(c2c(CC)c[nH]c2)=O)CC2CCC(C1)N2C(c1ccc(CO)o1)=O N1(C(=O)CC2CC23CC3)CCCC1C(=O)NCCOC(=O)C1CC1 N1(C(=O)CCCn2cccc2)CCC(C(=O)NC2CC=CCC2)(CO)C1 C#Cc1cnn(CC(=O)N(CC(=O)NC(C2CCOC2)C)C2CC2)c1 c1(OC)ccc(S(=O)(=O)Nc2ccc(SC#N)c(OC)c2)c(N(C)C)c1 Cc1cc(S(C)(=O)=O)ccc1CNC1CCC2(C1)CN(C(c1ncsc1C)=O)C2 N1(C(CCCCCC=C)=O)CCN(C(=O)CCCCC(C)=O)C2COCC12 c1(C(=O)NCC(CNC(C(C)OC)=O)O)csc(C)c1C C1(CN(C)NC)CCN(C(c2cccc(OCc3nnc(C)o3)c2)=O)CC1 c1(C(=O)NCC(CNC(c2c(CC)con2)=O)OC)ccc(-n2ccnn2)cc1 c1(OC)ccc(N)c(C(N2CC(OC)CC(NC(=O)CN(C)S(N)(=O)=O)C2)=O)c1 C(C)(CCCC(C)(C)C(C)(C)C)NC(C(n1cc(-c2cc(C)on2)nn1)C)=O C(=O)(CC(C)(C)CNC(C1CCOC(=O)CC1)=O)N(C)CCc1cccs1 c1(C(=O)NCC(CC)NC(=O)CCCCN(C)C)ncncc1Br C1(C(=O)NCCC(=C)CNC(c2nnc(O)nc2O)=O)CCS(=O)(=O)C12CCC2 N1(C(CC2CN(C)C2)=O)CC(N(C(=O)CN2CCC(C(N)=O)CC2)C)C(O)C1 C(CC(C)(O)CNC(=O)Cn1cc(CNC(=O)CC#N)nn1)OC CC(C)=C=CC(=O)N(C)CCC1CCN(C(=O)C=CC2CC2)CC1 N1(C(CC=CCC)=O)CCC(NC(=O)Cc2ccno2)C2(CCC2)C1 Cc1cc(F)c(C(=O)NC2CCC2NC(C2(C)CC=CC2)=O)cc1F CC1CC(NC(=O)CC2CCCCC2O)CN(C(=O)CCc2cnccn2)C1 Cc1ccc(NC(C2CC3CCC2N3C(=O)C(C2CCCCC2)O)=O)c(C)c1 C(C(CO)C(F)(F)F)NC(CCn1cc(-c2c(OCC)cc(C)s2)nn1)=O c1(C(=O)NCC2C(CNC(c3cc(C)oc3)=O)C2)cc2ccccc2c(=O)n1C N1(C(C=Cc2cn(C)nc2)=O)CCCOC(CCNC(c2nocc2Cl)=O)C1 c1(C(N(C2CCN(C(C(C)Cc3ccnn3C)=O)C2)C)=O)cc2n(n1)CCCO2 C(=O)(C(C(F)(F)F)C(F)(F)F)N(CCCc1noc(CNSC(C)C)n1)C c1(N2CCN(C(=O)CC)CC2)nc2c(c(=NCc3cccc(C)c3F)[nH]1)SCC2 C(CC(C(=O)N1CCCC(CSC)C1)NC(=O)C(C)OCC1CC1)SC N1(C(c2[nH]cc(CC)c2)=O)CC2(CCCC2NC(c2cn(C)nc2C)=O)C1 CN1CC(C(=O)NCC2CN(C(=O)Cc3ccc(F)cc3)CCO2)CCC1=O C1(CC)CCc2sc(C(N3CC(CNC(=O)C(C(C)C)OC)C3)=O)cc2C1 C(=O)(CCC(=O)N(CCCNC(c1cnc(C2CCCO2)s1)=O)CCC)OC C(=O)(C(C)(C1CCC1)NC(=O)CC1C=CCCC1)N(CCOC)CCOC C1(O)(C(C(=O)NCC2CCC2CO)F)CN(C(c2coc(C(F)F)n2)=O)C1 Cc1cc(Cl)cc(N)c1C(=O)NC(C)CNC(=O)CCOc1ccccc1Cl N1(C(C(CC)OC)=O)CCCC(CCO)(NC(=O)CC(C)C2CC2)C1 N1(C(C(=O)NN(CCC)C(N)=O)=O)CCCC(NC(=O)CCCOC(C)C)C1 CON1CC(C(N2CCC(C(=O)NCC(=O)NC3CCC3)C2)=O)CC1=O c1(C(=O)NC(Cn2cc(C(C(OC)OC)C)nn2)C)ccccc1CC#N C(=O)(C#CC1CC(F)(F)C1)NC1CCN(C(CS(N)(=O)=O)=O)C1C1CC1 CN1CC(C)(NC(=O)C(Cc2cnn(C)c2O)NC(=O)CCCSC)CCC1=O N1(C(c2ccc(C)o2)=O)CCN(C(=O)CCC2CC2CC)CC1CC1CC1 C1(C(=O)NC2CC(NC(c3ccc(Cl)o3)=O)C23CCC3)CCC2(CC1)OCCO2 c1(C(C)C)occc1C(N1CCC(OCCNC(C23CC(C)C2C3)=O)C1)=O c1(C(=O)NC2(C)CCCN(C(C3CCCC3C(F)F)=O)C2)ccnc2ncnn12 CC1CCn2cc(C(=O)NC3CC(CNC(=O)Cc4ccsc4)C3)nc2C1 N1(C(c2c(C)onc2CO)=O)CC2CC(NC(C3CCC(=O)N3C)=O)C2C1 C1(CNC(C(C)(C)COC2CC2)=O)CN(C(=O)CCC2CCOC2)C2(CCC2)C1 c1(COC)cccnc1C(N1CCC1CNC(=O)CSCCN(C)C)=O c1(NC(c2c3n(nc2)CC(C)CO3)=O)ccc(F)c2cnccc12 C=CCCC(C)(C)C(=O)NC1C2CN(C(=O)C(C)Cc3ccccc3)CC12 N1(C(c2c(C)cc(C)o2)=O)CCC(NC(c2ccc(C(C)C)c(F)c2)=O)C(F)C1 c1(C(N2CCCC(N(C)C(C3CC4(C3)CC43CC3)=O)C2)=O)c(F)cc(F)cc1Cl Cc1sc(=O)n(CC(N2CCC(O)(C(C)CNC(=O)C(C)(C)C#N)C2)=O)c1C CC1CN2CCN1CC2C(N1CC2CN(C=O)CC2C1)=O.C1CC2CCCC12 C(C(C)(C)CC(=O)N1CCOC(CNC(=O)CC2CSCCS2)C1)OC c1(C(N2C(C3CCN(C(=O)C=CC=C(Cl)Cl)C3)CCCC2)=O)nnc(O)nc1O C1(C(N(C2CC2CC(N2CCCC2CCC)=O)CC)=O)CC12CCCC2.CCO Cc1cc(C)n2c(CONCC3CCOC(C)(C)CN3)nnc2n1.c1(=O)c(=O)o1 C=C(CNCC1CC(OC(C)(C)C)C1)CCNC(=O)OC(C)(C)C CN1CCCCC1CNC(C1CNCCN1Cc1nccn1CC(F)(F)F)=O C=CC(C)(CC)C(=O)N1CC(O)(C2CCCN2C(c2cc(CC)ccc2C)=O)C1 N1(C(c2nc(CCC)oc2)=O)CCN(C(C2SCCS2)=O)C(C)CC1C C(=O)(C(C)(C)C1=CCN(C(=O)CCn2cncn2)C1)N1CCCC(C)(CO)C1 c1(NCCOC)cccc(CNC(=O)NC2(Cl)CC2(F)F)c1 C(C(CC(C)C)C(=O)N1CC(CC(=O)N(C)C)C12CCC2)OC CCCCC(O)C(=O)NC1CC(CNC(c2cnc(Cl)n2CC)=O)C(O)C1 N1(C(C=Cc2n(C)ccc2)=O)CCC2(CCN(C(C3CCCC(C)(C)C3)=O)C2)C1 C1(NC(C2(SC)CN(C(C3CCN(C)C3)=O)C2)=O)CCCCCC1F c1(C(N2CCCC(CCC)(NC(CCCCC)=O)C2)=O)ccc2cncn2c1 C1(C(=O)NCC2CCCC(NC(C3CCCN3C=O)=O)C2)(OC)CCSCC1 N1(C(C(C(C)(C)C)OC)=O)CCC2(CC1)C(NC(=O)CNC=O)CS2(=O)=O C1(CNC(C2CCOCC2)=O)CC2COCC2N1c1cnc(F)cn1 c1(C(=O)NC2CCCN(C(c3cc(C)ncc3)=O)CC2)coc2c(F)cccc12 c1(C(C)(C)C)ccc(C(N2CCN(C(=O)C(O)C3CC3)CC2)=O)cc1 C1(C(N2CC(C3CN(C(C(CC)C)=O)C3)C2)=O)CC2CCC(C1)C2(F)F c1(C(N2C(C(=O)NCC(C)(O)C3CC3)CCC2C2CC2)=O)cc2ncccc2[nH]1 C(CSc1ccccc1)(C(=O)NC(c1cn(C(C)(C)C)nn1)C)OC c1(C(N2C(CNC(c3n(CC)ccc3)=O)CC2)=O)ccc(C(=O)C2CC2)cc1 C#CCCC(=O)NCC(CC)NC(c1ccc(C2CCOC2)s1)=O c1(C(=O)NCCn2cncn2)cc[n+]([O-])cc1.C1CC(=O)N1C1CC1 C1(NC(C(C)=CC)=O)CCCC(CNC(=O)CSC)C1 C1(C(N)=O)(CNC(CCOCCC)=O)CN(C(=O)C(C)CC2CC2)C1 C12(C(=O)NCc3snc(C)n3)CC(CO1)N(C(c1scc(C)c1C)=O)C2 c1(C(=O)NCC2(C)CC(NC(c3ccsn3)=O)C2)ccc2ccccc2c1F N1(C(C2(CCOC)CCC2)=O)CCC2CCN(C(=O)CSC3CC3)C2C1 C12(CNC(C3(F)CCN(C(Cc4c(C)n[nH]c4C)=O)C3)=O)CCC(C1)C(=O)N2 C(CCC(=O)NC1CCN(C(C2CCOC2C(F)(F)F)=O)C1)N(C(C)=O)C C(=O)(N=c1[nH][nH]c2ncccc12)C1N(C(C2(C)CCC2)=O)CC=C1 CCC(CC)CC(=O)NCC1(CNC(=O)C(c2cc(F)cc(F)c2)C)CC1(F)F N1(C(C(C)CO)=O)C2CCCC1CC(NC(c1coc(C(N)=O)c1)=O)C2 Cc1cccc(F)c1C(N1CCC(CNC(=O)CCCC(C)C)C1)=O N#Cc1cn(CC(N2CC3CC(C2)N(C(c2cc(F)c[nH]2)=O)C3)=O)c(=O)nc1O N1(C(c2c(C)cc[nH]2)=O)CCOCC(F)(CNC(=O)C(C)Oc2cccnc2)C1 c1(NC2CCCN(C(CCC=C)=O)C2)ccc(C(=O)OC)cc1[N+](=O)[O-] N1(C(C(=O)NCC(CC#C)CC)=O)CC(CC2CCCCN2)c2ccccc21 c1(C(=O)NCC2C3CN(C(C(CC)=CC)=O)CC32)cc(=O)c(OC)cn1C C1(C(N)=O)(NC(C2CCC(CNC(C3CC(=O)C3)=O)C2)=O)CCCCC1 CCCS(=O)(=O)CC(=O)NC1(C2CN(C(=O)C(CC)OCC)C2)CC1 c1(NC(c2c(CNC(=O)CCC3CCC3)cco2)=O)cncc(F)c1 c1(C(=O)NCC2N(C(C=C(C)C3CC3)=O)CCC2C)cccc2cncn12 C1(C(=O)NC(C=C)C(F)(F)F)CN(C(=O)C(C)(C)CO)CC(C)O1 N#Cc1cccc(NC(=O)CN2CC3CC2CN3C(C2CC23CCSCC3)=O)c1 c1(C(=O)NCC2C(CNC(C(COC)COC)=O)C2)c(O)nnc2c1CCCC2 c1(NC(CC2CC(C)(C)N(C(c3cc(O)cs3)=O)C2)=O)ccc2c(c1)OCO2 C1(NC(C2CC(CCC)OCC2)=O)CCN(C(C2CC2CC)=O)C(C)C1 O=C(CS(=O)(=O)CC(F)(F)F)NCCC1CCCN(C(c2cnns2)=O)C1 N1(C(C(C)n2cncn2)=O)CCCC2CN(c3ncnc(Cl)c3F)CCC12 c1(C(=O)NC2(CNC(C3(F)CC3)=O)CCOCC2)cccc(C#CC2CC2)c1 CC(C)CC(O)C(C)C(=O)NCC#CCNC(c1cccnc1N(C)C)=O c1(OC)ccncc1C(=O)NC1(C)CCN(C(C2C=CCC2)=O)C1 CC1(CNC(c2n[nH]c(C3CC3)n2)=O)CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C1 CC1(C)CC2(CC2C(=O)NC(CNC(C2(n3cccn3)CC2)=O)CO)C1 C1(C(=O)NC(C2(O)CN(C(c3ccc(F)c(F)c3)=O)C2)C)CC2CCCC(C1)C2 N1(C(C(CN(CC)CC)F)=O)CCC(C)(C)C(NC(C2(C)CCCCC2)=O)C1 C#CCC(CC(F)F)C(=O)NC(COC)CNC(c1c(Cl)cnn1C)=O c1(OC)ccc(CC(N2CC3CC2(C(=O)O)CO3)=O)c2ccccc12 c1(C(N2C(C(N(C(C3CCOCC3)C)C)=O)C(C)C2)=O)ccc(O)c(F)c1 C1(CNC(c2nc(CC)oc2)=O)CN(C(=O)CSc2ccccc2Cl)CCCO1 N1(c2snc(C)n2)CCCOC(CNC(C23CC2COC3(C)C)=O)C1 c1(OCC=CC(=O)NC2CC2CNC(C2CCCCO2)=O)ccc(F)cc1 N1(C(Cn2c(C)nnn2)=O)CCC(N(C)C(c2c[nH]cc2C2CC2)=O)CC1 CC1(C)OCC2CC12C(=O)NCCNC(c1cc(-c2ccncc2)[nH]n1)=O C(=O)(CS(=O)(=O)C(C)C)NCC(CCOC)NC(C1C2CNC(=O)C12)=O c1(C(=O)N(CCC(F)F)CCO)cnn(CCNC(C2(C3CC3)CCCO2)=O)c1 c1(CC(=O)NC(C(=O)NCC2(CCC=C)CC2)C2(C)CC2)ccccn1 c1(C(=O)NCCC2(O)CN(C(CNC(N)=O)=O)C2)c[nH]c2ccc(F)cc2c1=O C1(C(N(C2CCCN(C(C(CC#C)C3CC3)=O)CC2)C)=O)C2CCC3C(C2)CC13 C#Cc1ccc(N)c(C(=O)NCC2(C)CCCN(C(C3CCC3(F)F)=O)C2)c1 C1(NC(=O)C(O)CN2CCCC2)CN(C(c2ccc[nH]2)=O)CC2(CC2)C1 C12(C(N(CC(=O)NCC3N(CC)CCCC3)C)=O)CCC(OC)C1CC2 CC(C)C(C(=O)NC(C)CCN(C)C(c1nc(-c2ccccn2)no1)=O)NC=O C1(CC(N2CCC(CO)(NC(C34C=CC(CC3)C4)=O)C2)=O)(COC)CCCCC1 N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(c2ccc(C)s2)=O)CC1C1CCC1 c1(OC)cncc(NC(C2CCN(Cc3cccc(-c4nn[nH]n4)c3)C2)=O)c1 CCCCS(=O)(=O)NC(C)C(N1CCC(NC(=O)C(CO)N(C)C)C1C)=O C1(C(NOCCCC)=O)(CN(C(C2(N3CCCC3)CC2)=O)CC)CC12CCC2 C(=O)(CCCC(C)C)N1CC(C(C(=O)NCC(CCC)OC)OC)C1 S(=O)(=O)(c1ccc(NC(=O)OC(C)(C)C)cc1F)N1C(C)(C)C(CO)CC1 n1(CC)ncc(C(N2CCCC(NC(c3ccc(CCO)cc3)=O)C2)=O)c1Cl N1(C(c2cnn(CC(F)F)c2)C(=O)NCCCC(=O)OCC)CCC(OC)C1 CC(CC(=O)N(C(C(=O)NC(C1CCC1)C1CCC1)C1CC1)C)n1cccc1 N1(C(c2cc(O)cc(F)c2)=O)CCCC2(C1)CN(C(C1(CO)CC(F)(F)C1)=O)C2 C(=O)(CCC[N+](=O)[O-])N1CCC(N(C)C(C2CCCS2)=O)C1 c1(CC)ccc(C(N2CCC(CN(C)C(C3CC3CC)=O)C2)=O)cc1[N+](=O)[O-] C1(NC(C(CCC)NC(N)=O)=O)CN(C(c2ccc(Cl)nn2)=O)CC2(CCC2)C1 C(=O)(C(C)CC(C)(C)C)NCCN(C(c1c(CC)cco1)=O)CCOC c1(C(N2CC(CCc3cn(CCC4CC4)nn3)C2)=O)ccc(C(=O)O)s1 Cc1cc(C(=O)NC2(C)CCN(C(=O)CN3CCCOCC3)CC2)cc(C)c1N n1(CCC)cc(C(C(=O)Nc2ccccc2)N(C2C3CCCC23)C)cn1 N1(C(C(C)OCC=C)=O)CC2CC(C1)C2NC(=O)C(F)C1CC1 Cn1nnc2c(C(=O)Nc3cncc(C(C)(C)F)c3)cccc12 C1(C(N2CCC(NC(C3CCN(C)C3)=O)C2)=O)CC12CCOCC2 c1(CNC(C2CCN(C(C3(C)C(C)CCC3)=O)CC2)=O)c[nH]c2ccccc12 CC(CNC(=O)C(C1CC1)C1CC1)C(=O)N1CC(O)(c2nn[nH]n2)C1 Cc1cnn(CC(=O)NCC2(O)CC(C(=O)NC(c3ccc(C)s3)C)C2)c1 N1(C(c2nc(C)on2)C)CCC2(CN(C(=O)Cn3ncnn3)CC(C)O2)C1 N1(C(C2C(C(=O)OC)CCO2)=O)CC2(CNC(c3ccc(O)nn3)=O)CC1CO2 c1(C(N(CC(C)NC(c2c(CCC)occ2)=O)C)=O)nc(Br)cn1C(C)C N1(C(C(CC=C)CNc2cc(O)ncn2)=O)CCC(C2CC2)C1C(=O)NC N1(C(c2c(C)cno2)=O)CCC(C)(C)C(NC(C2CC3CCC2C3)=O)C1 C(CCC(=O)NC(C(=O)N(C)CCN1CCCC1=O)C1(O)CCC1)OC C(CCC(=O)N(C(C)CO)C)(C(C)C)NC(c1c(CC)nccn1)=O CN1CCC(NC(C2CC2NC(=O)Nc2ccc(N(C)C)cc2)=O)CC1 c1(OC)c(F)cc(C(N2CC(NC(=O)CC(C)F)C(N=[N+]=[N-])C2)=O)cc1Br CN(C(=NCCCc1cccs1)NCC1CCOC1)CC1CCCCC1 C#Cc1ccc(C(N2CCN(C(=O)Cn3ncc(Cl)c3C)C3CC23)=O)cc1Cl C(c1ccnc(O)c1)=CC(N1CCC1CNC(c1ccn(C2CCCC2)n1)=O)=O C=C(Cl)C(C)(C)C(=O)NCCC(C)NC(c1cnn(-c2ccc(O)nn2)c1C)=O CC1CCc2[nH]c(C(=O)NCC3CC3NC(c3cc(Cl)ccc3O)=O)cc2C1 N1(C(CCC(=C)Cl)=O)CCN(C(=O)C(F)(F)C2CC2)CC1CC1CC1 N1(C(C(F)=CC)=O)CC2CCOC2(CNC(c2cn3ccccc3n2)=O)C1 c1(CC(=O)NC2(CCCNC(c3cc(C)on3)=O)CC2)ccc2sccc2c1 c1(C(=O)NCCN(C)C(c2ccc(Br)cc2Cl)=O)ccc(O)c(N)n1 O=C(Cc1csc(=NCc2cc(Br)cc3[nH]ncc23)[nH]1)N=c1ccnc(Br)[nH]1 N1(C(CCNS(CC)(=O)=O)=O)CCC(O)(CN(C(=O)C=CC(F)(F)F)C)C1 C1(O)(CCNC(C=CC(C)C)=O)CCCN(C(=O)Cc2ccccc2C#N)C1 C12(NC(C=CCOC)=O)CCCCC1CN(C(c1cccn3nnnc13)=O)C2 Cc1onc(CC(=O)NCC2CCC(NC(=O)C=C3CCC(C)C3)CC2)c1C#N N#Cc1cccc2[nH]c(C(=O)NCC3CCC3NC(c3cc(CO)[nH]n3)=O)cc12 C(=O)(C(O)CNC(c1occc1C1CC1)=O)NCC(C1CC1)OC c1(CN(C(CCC2C(C)C2)C(=O)N2CCCNCC2)C)cccc(F)c1F C#Cc1ccc(C(N2CC(CNC(c3cncc(Cl)c3)=O)C(O)C2)=O)c(C)c1 C1(C(N2CCCN(C(=O)Cc3cscn3)C(CO)C2)=O)CC2CSCC(C1)C2 Cc1ccc(C#N)cc1C(=O)NC1(C(=O)NCC2CC2Cl)CC(O)C1 CC(C)C(C)(O)C(=O)NCc1ccoc1C(=O)N(C)C(C)C1CC1 CCC(C(=O)NC(C)CCN(C)Cc1cc(-c2cccs2)on1)OC c1(C(N(C2C(SC)CCC2)C)=O)ccc(C(=O)O)c(P(C)(C)=O)c1 C1(OC)CCC(C2CC2)C1.C1(CC(=O)CNC=O)(C(=O)NCCCNC)CCC1 c1(C(=O)NC2(C)CCN(C(c3c(C)onc3Cl)=O)C2)cc2c(Cl)nccc2o1 C12(NC(CC(=O)OCC)=O)CCOCC1CN(C(c1cnc(Br)c(C)c1)=O)C2 N1(C(c2c(C)nc(C(C)C)o2)=O)CCC2CC2(NC(=O)COC(F)F)CC1 Cn1cnc(C(=O)NC2CCCN(C(=O)OC(C)(C)C)CC2)cc1=O c1(-c2n(CCC)nc(CCCO)n2)ccc(OC)c(-c2ccccn2)c1 c1(CC#N)cccc(C(=O)NC2CCOC2C(=O)NC(CO)CCO)c1 Fc1cc(-c2nc(-c3ccoc3)nn2CC(F)F)ccc1Cl c1(N2C(C)CC(NC(c3ccc4c(c3)CCOC4)=O)C2)ccc(Cl)cc1[N+](=O)[O-] Cc1noc(C)c1C(=O)NCCC1CC(C(=O)NC2(CCO)CCC2)C1 c1(OC)cc(F)ccc1C(=O)NC(C)CCCNC(=O)Cc1cccc(SC)c1 CCCC(C(=O)NC1CCN(C(C2(CCCOC)CN(C)C2)=O)C1)OCC C1(C(=O)NC(C)Cn2nccn2)(OC)CCN(C(C2(C3CC3)CC2)=O)C1 C(=O)(C(F)(F)C(O)CC)OCCCN1CCCC(NC(=O)OC(C)(C)C)C1=O c1(CN2CC(=O)N(CCC(F)(F)F)NC2=O)cc(C(=O)O)c2n1CCCC2 CC(C)(CCNC(=O)C=CBr)NC(c1ccccn1)=O c1(CC(N2CC(NC(=O)Cc3ccnc(Br)c3)C(O)C2)=O)cc(F)c(F)cc1F CCCS(=O)(=O)C(C)C(=O)NCC(C(C)C)NC(c1cnn2ccsc12)=O c1(C(N2C(C)C(NC(=O)C=C(C3CC3)C3CC3)CCC2)=O)ccc2c(c1)CCO2 N12CCCC1C(NCCO)C2=O.n1(CSC)cc(NC(S(C)(=O)=O)C2CC2)nn1 C(C(N=[N+]=[N-])C(=O)N1CCC(NC(C2CCCO2)=O)C1(C)C)OCC C(C(=O)NC(C)C(C)(C)NC(=O)Cc1cncc(F)c1)(C(C)(C)C)SC c1(OC(CC)C(=O)N(C2CCN(C(c3ccc[nH]3)=O)C2)CCO)ccccc1F CC1C(NC(c2n[nH]c(O)n2)=O)CC2CCC1N2C(c1ccc2c(c1)CC2)=O c1(C(=O)NCC2N(C(C=CCOCCOC)=O)CC2)cccc(OC)c1Cl C1(NC(c2cscn2)=O)Cc2ccccc2C1NC(c1cccc(F)c1O)=O C1(NC(C=CCOC)=O)CCN(C(=O)C(C2CCCN(C)C2)(C)C)CCC1CO N1(Cc2[nH]nc(C(=O)OCC)n2)CCc2nc(Cl)cc(Cl)c2C1 C1(CNC(CS(CC)=O)=O)CN(C(=O)CN2CC(OC)C2)CC1(C)C N1(C(C(C)N(C)C(c2ncccc2Cl)=O)=O)CCN(C)CC(O)C1 N1(C(c2cc(SC)oc2C)=O)CC2CC1CC2NC(c1sccc1Cl)=O CCCC(CNC(=O)Cc1cscn1)C(=O)NC1CCC(C(N)=O)C1 C12(C(=O)NC(C)(C)CNC(=O)CC3CCOCC3)CCCC1OCC2 c1(-c2ccc(OC)cc2CN(CCCCO)C)cc(F)c(F)cc1C CC(C)CC(C(=O)N1CC(O)(CNC(C2CC3CCC2CC3)=O)C1)n1ccnc1 O=C(C1=NN(CCO)C(=O)CC1)NCC12CC1CN(C(c1ccncc1F)=O)C2 c1(CCNC(=O)NCCN2CC(C)OC(C)C2)ccc2c(c1)OC(F)(F)O2 C1(C(=O)NC(C2CCCC2)CO)(OC)CCN(C(C2CC(O)C(F)C2)=O)C1 C1(CNC(C(n2ncc(C)c2)C)=O)CCCN(C(c2cnc(N)c(Cl)c2)=O)CC1 C1(C(=O)NC2CCN(C(=O)OC(C)(C)C)C2(C)C)CCC2(CCC2)O1 C(C(=O)N1CCC(C(=O)Nc2cccc(CCO)c2)O1)c1cnc(C)s1 N1(C(C2(C(CC)=O)CC2)=O)CC2(CO)CC1(C(=O)NCC(F)Cl)C2 c1(C(=O)OCC)ccc(C(N2CCC(NC(=O)CC3CC3)C(O)C2)=O)cc1O C(=O)(CCC(C)(C)C)NC(CNC(COC(CC)(C)C)=O)C(C)C Cc1nccc(C(=O)NC(C)(C)C(C)NC(=O)CCc2cc(F)cc(F)c2)c1C c1(SCC(=O)Nc2nnc(-c3cncc(C(F)(F)F)c3)s2)ccc2c(c1)CCO2 Cc1cc(C(=O)NCC2CN(C(=O)CCCC3CC3)C(C)(C)C2)cc2ccsc12 c1(SC)ccc(N)cc1C(=O)NC(C)(CNC(c1oc(C(F)F)cc1C)=O)CO CC1CCCC(CC(=O)NCC(O)CNC(=O)C(O)C2CCCC2)O1 C#Cc1cc(F)c(C(N2CC(NC(c3occ4c3CCC4)=O)C(C)C2)=O)cc1F CCCC(C(=O)N1CC2(C)CC1(C(=O)NC1(C)CCOC1=O)C2)C(C)C C1(C(=O)NCCS(Cc2n(CCCC)ncc2)(=O)=O)CCN(S(=O)(=O)N(C)C)CC1 C1(NC(c2cc(C(CC)C)no2)=O)CN(C(c2c(C)ccn2C)=O)CC1N=[N+]=[N-] CC(C)(C)C(C#N)C(=O)N1CC2(C(N3CC(=O)NC4(CC4)C3)=O)CC1CCO2 C1(NC(C2(CCC)CCNC2=O)=O)CCC2(CC1)CN(C(c1ccsc1C)=O)C2 C1(NC(=O)CC2CC(C(F)F)C2)CCC2CCN(C(C3CCCCO3)=O)C12 n1(CCCC)nnnc1C(C1CC1)NC1COC(C(F)F)C1 C(=O)(CCCC(=O)NCC1C(C)CCN1C(=O)CN(c1ncccn1)C)NCC C1(O)(CNC(CC=CC)=O)CC(NC(=O)C(C)(C)OC(C)=O)C1 c1(OC)ccc(OC)c(C=CC(=O)NC2(CNC(=O)CC3CC4(CC4)C3)CCC2)c1 c1(SCC)c[nH]c2nc[nH]c(=NCC(CO)C3CCCCC3)c12 N1(C(N)=O)CCC(NC(=O)CC2CCCC(NC(=O)CCNC(=O)CO)C2)CC1 Cc1ccc(F)c(C(N2CCCC2CNC(C2(CO)CCCCO2)=O)=O)c1 C1(C(C)NC(c2cnn(CC)n2)=O)CCCCN1C(c1occc1C)=O c1ccc2c(c1)OCC21CN(c2nc(-c3ccccc3)nc(=N)[nH]2)C1 Nc1cc(F)c(Cl)cc1C(=O)NC1(CCNC(=O)C(F)CC2CC2)CCCC1 C1(OC)(CNn2cc(-c3cc(F)cc(C)c3N)nn2)CC(C)CC(C)C1 N1(C(C(C#C)(C)C)=O)CCC(C2CCN(C(=O)CC34CCCC3C4)C2)CC1 CCC(Cc1ccccc1)C(=O)N1CC2CC2(NC(c2ccncc2C)=O)C1 c1(C(=O)NC2(CCOC)CCN(C(C(CC)C(C)O)=O)C2)nc2ncccn2n1 Cc1cc(C(=O)NC(CC2CC2)C(=O)NCCOCCN=[N+]=[N-])nc(O)n1 N1(C(C(COC)N(C)C)=O)CC(C(N2CCC23CCCCC3)=O)CC12CCC2 CN1CC2(CC2)CC1C(N1CC(C2CC2C(N2CCCC2C(O)CO)=O)C1)=O CC1CN(c2nnc(CC(F)(F)F)s2)CCC1NC(=O)Cc1c(O)ncnc1O N1(C(CC(CC)C)=O)CC(NC(=O)C(C)(O)C(F)(F)F)Cc2ccccc21 C=CCC(CC(F)F)C(=O)NCC1C2CN(C(c3ncc(N)cc3Cl)=O)CC12 C(=O)(C#CC1(C)COC1)N1C(CC(=O)NC2(CC=C)CCCCC2)CCCC1 CN1CC(NC(C2COCCC2NC(=O)C(O)C(F)(F)F)=O)CCC1=O N1(C(C=Cc2c(C)cncc2)=O)CCC2(CCC2NC(c2nccn2C)=O)CC1 c1(NC(CC(C)(CO)NC(=O)CCOC2CC2)=O)ccc(C(F)(F)C(F)F)cc1 N1(C(C)=O)CCC(S(=O)(=O)NC(c2cc(F)cc(F)c2F)=O)CC1 N1(C(C(CC(=C)C)OC)=O)CCCN(C(c2ccc(F)cc2OC)=O)CC1C c1(C(=O)NC(C2CN(C(CCOC(C)C)=O)C2)C)cn(C2CC2)nn1 N1(C(c2cn(CCNC(c3ncccn3)=O)nc2)=O)CCC(O)(CC2CC2)C1 N1(C(CC=CCC)=O)CCC2(CCN(C(=O)C(C)OC)CC2)C1 c1(NC(C(C)CNC(c2cncn2C)=O)=O)cccc([N+](=O)[O-])c1 N1(C(C(C(C)C)=O)=O)CC(NC(=O)CSC2CCCCO2)CCC(O)C1 Cc1scc(C(=O)NC2(CCNC(=O)CO)CC2)c1N c1(C(N2CC(NC(c3ccc(C4C(C)C4)o3)=O)C2)=O)cnc(C2CCC2)nc1O N1(C(C(CNC(=O)Cc2ncoc2C)OC)=O)CCN2CC(O)CC2C1 c1(CC(=O)NCCC2CN(C(C(C)O)=O)CC2C)ccc2ccccc2c1 c1(C(=O)NC(CN(C(c2c(CCC)nco2)=O)C)CC)ccc2nc(O)[nH]c2n1 C1(C(=O)NC2CN(C(c3cc(COC)sc3)=O)CC2F)CC2CCC(C1)O2 c1(C(=O)NCC2N(C(C3(OC)CC3)=O)CC2)c(Br)ccc(F)c1C N1(C(CC2CC(C)C2)=O)CCC2(CCCN2C(C2CCC(C)(C)OC2)=O)C1 Cc1ccc2c(C(N3CCC(CNC(C4(F)CC4C)=O)C34CCC4)=O)csc2c1 C1(C(N(C)CC2CCCN2C(C2(C#N)CC2(C)C)=O)=O)CC2(CCCC2)CO1 c1(C(=O)NCCCCCNC(C(C)OC(C)(C)C)=O)cccc(Br)c1F CCC(C(=O)NC1CC1CNC(=O)CCOC)OC1CCCCC1 N1(C(c2ccc(OC)nn2)=O)CC(C2CCCN(C(c3n[nH]cc3C)=O)C2)C1 Cc1cc(C(=O)NCC2CN(C(C3CSC3)=O)CCO2)c(C)n1NC(N)=O C1(C(N(C)CC2N(C(c3cn(C(C)C)nc3)=O)CCC2)=O)CCCC2C1C2(F)F N1(C(c2c(C)nc(C)[nH]2)=O)CCC2(CCC2NC(C2CCCCC2(C)C)=O)CC1 C1(NC(CCNC(C2CC3(CCC3)CO2)=O)=O)CCCCCC1F c1(-n2c(Cc3ccccc3)nc(C(C)C3CC3)n2)ccc(Cl)cc1Br Cc1sc(C)c(C(=O)NC2CC(O)(CNC(=O)C(C)C3CCCC3)C2)c1C#N C1(C(=O)NCC(CNC(c2nc(C)oc2)=O)CO)CCN(C2CC2)S1(=O)=O c1(C(N2CCC(CN(C(=O)C=CC3CC3)C)C2)=O)cccc2ccc(O)nc12 c1(OC)ncc(-c2cn(C3CCN(C(=O)Cc4n[nH]c(C)n4)C3)nn2)cc1F C12(CCNC(C(C=CC)O)=O)CCC(CC1)N(C(=O)CCc1cc(F)ccn1)C2 C(N=c1cc(NCCC(C)CC(C)C)nc[nH]1)c1cc(OC)c(OC)cc1 CCC(CC(C)C)C(=O)NC(C)(CO)C(=O)N1CCN(C(C)(C)C)CC1 N#Cc1ccc(CC(N2CCC3(C2)CN(C(C2CCC(=O)NC2)=O)C3)=O)c(F)c1 c1(C(=O)NC2(CNC(CCc3cc(C)on3)=O)CCOCC2)ncc(Cl)nc1Cl c1(C(=O)NCCN(CCOC)C(C2(C)CC2)=O)cc(F)cc2nn(C)cc12 C(C(C)(C)C(=O)NCC12CC(CSC)(CO1)C2)N(C)C(c1ncc[nH]c1=O)=O N1(C(CC2N(C(C3CCC(C)(CC)O3)=O)CCOC2)=O)CCC2(CCO2)C1 c1(NCC)cccc(C(=O)NCCNC(c2cc(CCOC)on2)=O)c1 c1(NC(C(CCCOC)NC(=O)C=C=C(C)C)=O)cccc2cnc(Cl)cc12 C(=O)(C(C)(C)CC(=O)OC)NCC(CC)NC(=O)C(C(C)(C)C)NC(C)=O C1(NC(C(CCC)NC(C)=O)=O)CC2CCCC(C1)N2C(=O)C(Cl)=CCl C1(C(=O)NC(C)CN2CCOCC2)CN(C(c2cncc(Cl)c2)=O)CC1C(C)C C1(CNC(CN(CCCCCC)C)=O)COCCN(C(=O)C(C)=O)C1 C1(C(=O)NC2CCN(C(c3cc(CO)on3)=O)C2C)(OC)CCCOC1 N1(C(c2c(C(C)(C)C)n[nH]c2)=O)CCC2(CC1)CC2NC(=O)CCc1cncs1 N1(C(c2c(C)nc(COC)s2)=O)CC=C(C(=O)O)CC1 CN1CC(O)CCC1C(=O)NCC1CCN(C(c2ccc(O)cc2F)=O)C1 c1(C(N(C(C)CNC(c2cnnn2C)=O)C)=O)cnn2c1CC(C)CC2 Cc1cccc(OC(c2ccc(NC(C3CC4CCC34)=O)cc2)C)n1 Cc1cn2c(n1)CN(C(=O)CCC(C)(C)NC(=O)CS(C)(=O)=O)CC2 N1(C(Cn2c(C)cnc2)=O)CCOC(CNC(=O)CCS(C)=O)C1 c1(C(=O)NCC(C)(C2CC2)NC(=O)CCCC2CCCC2)cc(C(F)(F)F)no1 CC(C)CC(C(=O)NC1CC(CNC(C2CC2c2nccn2C)=O)C1)C(N)=O CC1CN(C(C2CCC(O)CN2C(=O)Cc2cncn2C)=O)CC2(CCC2)O1 c1(C(=O)OCC(N2CC(C)C(O)CC2)=O)c(N)cc(Cl)nc1Cl C1(C(N(CCOC)CCNC(=O)Cc2ccsc2C)=O)CCN(C(N)=O)CC1 Cc1nc(Cl)cc(=NCC2CCCC(NC(c3ccc(-c4cc[nH]n4)s3)=O)C2)[nH]1 N1(C(c2c(CC)nns2)=O)CCC(O)(C(C)NC(c2nn(C)nc2C)=O)C1 C(c1cn(C2CC(NC(c3ccc(C4CC4C)cc3)=O)C2)nn1)=CC C1(C2CC2)(NC(C=CC(=O)NC2CC2)=O)CCN(C(=O)C(c2cccnc2)O)C1 c1(C(N2CCN(C(C(CC)N(C)C)=O)CC2C)=O)cc2cc(C)ccc2nc1C N1(C(C2(SC)CC(O)C2)=O)CCC(C)N(C(=O)C(c2ccccc2)SC)CC1 CN1C(=O)CCCC1C(=O)NCC1(C(=O)NCC2(NC)CC3CCCC23)CCC1 C1(C(=O)NCc2c(CNC(C3=NOC(C)C3)=O)cccc2)COCC2(CCC2)O1 N1(C(C2OCCN(C(C3CCC(C(N)=O)C3)=O)CC2)=O)CC2CCOC(=O)C2C1 Cc1cc(C(=O)NCCNC(C2CCN(S(N)(=O)=O)CC2)=O)c2cnn(C)c2n1 C=C1CC(C)(C(=O)NC(C2CCCCC2)C(C)NC(=O)CC2CCCC2)C1 c1(C(=O)NCC(CNC(c2c(CC)con2)=O)C)c[nH]c2ncc(Br)cc12 C12(CNC(CCC=C)=O)CCC(CC1)N2C(=O)Cc1c(C)nn(C(F)F)c1C C1(C(=O)NCCCCCNC(C2CCC(C)(C)C2)=O)CCC(F)(F)CO1 C(=O)(CCCC(N)=O)N1CC(NC(CCc2cn(C)nc2)=O)C(O)C1 C1(NC(C2N(C(CCOCCC)=O)CCC2)=O)CC12CCOCC2 C(=O)(CCC(F)(F)Cn1cncn1)NC1CN(C(c2cc(=N)[nH]cc2Br)=O)C1 N1(C(C(C)SC)=O)CC2(C)CC1(C(=O)Nc1ccc(OCCO)cc1)C2 C=CCCCC(=O)N1CC(CC(C)NC(c2sncc2C)=O)C1 CN1CCC(C)(C(=O)NCC2CCN(C(=O)CC3CCC(C(F)(F)F)O3)C2)C1=O Cc1sc(C(=O)NC2CC2NC(c2cc(C(C)C)on2)=O)cc1Br N1(C(C)=O)CCCCC1C(C)(C)CN(C(C1CC1c1cncn1C)=O)C1CC1 CN1CCN(C(=O)C(F)C(C)(F)F)CC1C(=O)NCCc1cccc(F)n1 N1(C(c2c(C)cncc2C)=O)CCC(CC(=O)CC2CCCC2)C(C)(C)C1 c1(NC(=O)CNC(=O)N(c2ccccc2)CCCn2cncn2)ccccc1 c1(SC)cc(N2CCOC(CNC(=O)C(c3cccc(C)c3)O)C2)nc(SC)n1 c1(C(=O)NCC#CCCO)ccc(F)c([N+](=O)[O-])c1 C1(C)(COC)CCN(C(=NCCC2(O)CCCOC2)NCCCCl)CC1 c1(C(=O)NCC2CC(F)(CNC(c3c(CC)nns3)=O)C2)cc(C#N)ccc1F c1(OC)cc2c(cc1C(N1C(C)C3CC1C3NC(=O)C(C)(C)C(C)C)=O)OCO2 C1(CC)CCCC(c2nnnn2CC2CC2)(NCCCN2C(=O)CCCC2=O)C1 c1(CC)cccc(C(=O)NCC2CCN2C(c2cc(C(N)=O)co2)=O)c1 C(CCCO)N(C(CN(C(=O)C(C)C1CCCO1)CC(C)C)=O)C C(=O)(CCCCN=[N+]=[N-])NCC(CC(=O)NCC(C)(CO)CO)OC c1(OCC)cc2ccc1ONC1CCN(CC1)CC(=O)N2.C(C(C)C)NC C1(SCC(=O)NCC=CCNC(=O)CCc2cocn2)CCOC1=O C1(NC(CCC=C(C)C)=O)CN(C(=O)CC2CN(C)C2)CC1c1ccccc1F N1(C(COC(CC)CC)=O)CCOCC1CNC(=O)CCc1cccnc1 C1(CNC(C2(Oc3ccc(CC)cc3)CC2)=O)CC2(C(C=O)CC)CN1C(=O)C2 C(=O)(C1=COCC1)N(CCN(C(C1CC1(C)C)=O)CC)CC c1(NC(N2CCCCC2n2cc(-c3c(C)scc3)nn2)=O)nn(C)c(Br)c1C CC(C)(C)CCCCC(=O)N1CC2CC1C2NC(C1(C)COC(=O)OC1)=O c1(C(N2CCN(C(c3n(CC)ccc3)=O)C3C2C3)=O)ccnc(S(N)(=O)=O)c1 CCC(C)C(C(=O)NCCC1(NC(c2ccn(C(C)C)n2)=O)CC1)OC CC1(C)CCCCC1C(=O)NCCNC(c1cc(Cl)no1)=O c1(C(N(CCC(C)O)C)=O)cc(CNC(=O)C=CCN2CCC2)[nH]n1 N1(C(CC2CNC(=O)O2)=O)CC=C(C(=O)NC2CC3(CCC3)C2O)CC1 C=CCC(CNC(=O)CCc1cnc(C)o1)NC(c1cc(C2CCOC2)[nH]n1)=O N1(C(c2nc(OC)c(F)cn2)=O)CC2CC(NC(C3CCCN3C=O)=O)CC1C2 N1(C(CSc2n(C)ncc2)=O)CCCC2CN(C(C3(C)CC(F)(F)C3)=O)CCC12 C(=O)(C(CO)C(C)(C)C)NCc1cncc(C(N2CCOCC(=C)C2)=O)c1 c1(CC(=O)NC2CCCN(C(c3c(O)nc(C)s3)=O)C2)ccc2ccoc2c1 CCC(CC(=O)N1CC2C(CO)C2C1)N(C(=O)CCC(C)N(C)C)C c1(C(=O)NC2CC(NC(Cc3c(C)con3)=O)C23CCC3)cncc([N+](=O)[O-])c1 c1(CNC(CCCOCC=C)=O)cnn(C)c1C(=O)NCC1CC(CO)CO1 N1(C(C(Cc2c(C)nn(C)c2C)C)=O)CC(C)CN(C(=O)CC2CSC2)C(C)C1 c1(C(=O)NCc2n(C)c(Cl)cn2)cc(=NC2C=CCC2)[nH]c(=N)[nH]1 C1(C)(CCNC(C(CC)F)=O)CCN(C(c2ccc(C(C)C)cn2)=O)CC1 c1(C(=O)NCC(C)(C2CC2)NC(c2cscn2)=O)ccc(C2COC2)cc1 C1(OC)(CNC(c2cnc(CC3CC3)s2)=O)CCN(C(=O)CCCCO)CC1 CC1(C)CC1(C#N)C(N1CCOC(CCCNC(=O)CC(Cl)Cl)C1)=O C1(CNC(C2CCC(=O)N2)=O)CC2CCC1N2C(=O)C(c1ccc(F)cc1F)=O C#CC1(C(=O)NC2CC(C)N(C(=O)Cc3c(F)cccc3Cl)C2)CCOCC1 N1(C(c2cc(C)cc(O)c2)=O)CCC(C)N(C(=O)CC(C)(C)N(C)C)CC1 S(=O)(=O)(c1c(OC)cccc1F)N1CC2CN(C(CC(=O)NCC)=O)CC2C1 CC1CN(C(=O)COC2CCC2)CC(C)C1NC(c1snc2ccccc12)=O N1(c2snc(C(C)SC)n2)CCCC(C(=O)OC)C1 CC1(O)CCN(C(=O)CC2CCC(NC(C3C4CC5C(C4)C35)=O)C2)CC1 c1(OCC(=O)NCC2(F)CN(C(c3nc(C4CC4)cs3)=O)C2)cccc(O)c1.OCO CCCC(CCC)C(=O)NCc1ccc(C(N2CC(CO)C(O)C2)=O)cc1 C#CC1(C(=O)NCCNC(C)=O)CCN(C(=O)C=C2CCC(C)CC2)C1 c1(C(=O)NCCN(C)C(C2CCCN2C=O)=O)cc(F)c(Cl)c([N+](=O)[O-])c1Cl C(=O)(C1=Cc2cccc(Br)c2OC1)NCCCC(C)NC(=O)C1=CCC1 O=C(CCCC1CCC1)Nc1ccsc1I c1(C(=O)NC2CC(NC(C(CC)C)=O)C(O)C2)ccc2nc[nH]c2n1 c1(C(N2CC(O)(CNC(Cc3c(C)nc(Cl)cc3)=O)C2)=O)cccc2c1COC2 C1(NC(=NC)NCC2(C3(CC)CCCCCC3)CC2)CCOC2(CCOCC2)C1 C1(CC)(NC(C2CCSC2)=O)CCCN(C(c2ccc(C(=O)OC)nc2)=O)C1 C(=O)(CCCC(=O)N(C)C)N1CCC(NC(COCc2c(C)ncs2)=O)C1C c1(C(N(C)C)=O)ccc(NC(C2CCC3CC23)=O)cn1 N1(CCOCCOCC)C2CCC1CN(C(=O)Cc1cnnn1C)C2 Cc1c[nH]c2ncnc(N3CC4CN(C(c5ccccc5CO)=O)C4C3)c12 c1(C(=O)NCC(C)NC(CCOCCCOC)=O)ccc2c(c1)OCCNC2=O N1(C(CCNC(=O)OC)=O)CC2CC1(CNC(=O)CC1CCCN(C)C1)C2 Cc1nc2c(o1)CCN(C(C13CC1CN(C(c1sc(Br)nc1C)=O)C3)=O)C2 C(C)(C(C(=O)NC(C(=O)NC1CCOCC1F)C1CCC1)N(C)C)OC C(=O)(CC(C(C)C)NC(=O)C1CC1)NC(CC1CN(C(CCC=C(C)C)=O)C1)C CCCCC(F)C(=O)N1CCCC(CCNC(c2cnn(CC)c2)=O)C1 Cc1cc(C(=O)NC2CN(S(=O)(=O)CC3CC3)CC2(F)F)ccc1F c1(NC(C(N2CCCC(n3ccc(C)n3)C2)C)=O)cccc(Cl)c1C C(=O)(C1(C)CCCc2ccccc21)NCCC(C)(C)NC(C(F)=CCC)=O C(CCCCC(=O)N1CCC(c2nn[nH]n2)C1)N(C(c1cc(C)ncc1)=O)C C1(F)(CNC(C(CC)(C)O)=O)CCCN(C(=O)COc2ccc(C)c(C)c2)C1 Cc1ccc2oc(C(N3CCC(C)C3CNC(C3(C)CCCO3)=O)=O)cc2c1 c1(CNc2cnn(-c3cc(C)cc(C)c3)n2)nc2c(s1)CC(C(C)(C)C)CC2 c1(CC(=O)NC23C(CN(C(C4(N(C)C)CC4)=O)C2)C3)ccc(F)cc1[N+](=O)[O-] C(=O)(C(C)(C)CC(=O)NCCNC(=O)CC(C(F)F)c1ccc(F)cc1Cl)OC C1(CCCCNC(COCCCSC)=O)CCCCN1C(=O)C(CC)N(C)C C1(N(C(=O)CC(C)(C)C)C)CCC2CN(C(=O)Cn3ccnc3)CC12 C(F)(c1ccccc1)=CC(=O)N(CCCNC(CCSCC(C)C)=O)CCO c1(C(=O)OC)cc(NC(=O)CCCSC)cc(NC(C2CCCOC2)=O)c1C O=C(N=c1nc2cc(Br)ccn2[nH]1)N1Cc2ccncc2C(F)(F)C1 C1(CC)C(NC(C23COC(CF)(C2)C3)=O)CCCN1C(c1ncsc1C)=O N(C1CCCc2nc(-c3cn(C(C)COC)nn3)sc21)CC.C(C(=O)OC)O C1(CC(=O)NCC2(C(N)=O)CN(C(C3CCN3C(C)(C)C)=O)C2)CN2CCN1CC2 c1(CNC(CC2(CCC=C)CC2)=O)ccc(C(=O)NCC(O)C(N)=O)cn1 N1(C(C2C(C)(COC)C2)=O)CCC2CCN(C(=O)CC3CC(OC)C3)C2C1 c1(C(C)C)ccc(C(C)C(=O)NCc2csc(-c3ccccc3)n2)cc1 N1(C(COCCC)=O)CCCC1CNCC1CCC1(C)C C1(N(C(=O)C(C)(C)C)C)CCC2(CC1)CC2NC(=O)C(=O)NCC(F)F c1(C(N(C2CC2)CC2N(C(COCCCC#C)=O)CCC2)=O)cc2[nH]ccc2s1 c1(OC)ccc(F)c(N)c1C(N1CCC(C)N(C(=O)Cn2nnc(C)n2)CC1)=O c1(CNC(C2CC2Cl)=O)n[nH]c2c1CN(C(c1c[nH]c3cccnc13)=O)CC2 N1C(=S)NC(C(C)(C)C(F)(F)F)C2=C1CC1(CCC1)NC2=O.C1CCNCC1 N1(CCN(C)C(C2CN(C(=O)NC(C)C)C2)=O)CCCCC1 C(CCC(CCC)NC(C1CC12CCC2)=O)NC(CCCC#C)=O N1(C(C2(CSC)CC2)=O)CC(C(C)NC(=O)CC2CC2(Cl)Cl)C1 Cc1ccc(Cl)c(C(=O)NCCC2(C)CCN(C(=O)C(C)NC(C)(C)C)C2)c1N C=CCCC(C(=O)N1CC(C#N)C1)NC(=O)CC1CCCC12CC2 N1(C(C2C(C(=O)OCC)C2)=O)CCN(C(=O)C(C)(C)C(C)C)C(C)C1 N1(C(Cc2c(C)ccs2)=O)CCC2C1CCN2C(C1CC1c1ccccc1)=O O=C(CC(F)(F)C(F)(F)F)N1CCCC(n2cc(CO)nn2)C1 c1(NC(C2CC2NCc2ccc([N+](=O)[O-])cn2)=O)ccc(I)cc1[N+](=O)[O-] c1(NC2CCN(C(=O)NC3CCCC(n4c(=N)nc[nH]4)C3)C2)cc(F)cc(F)c1 Cc1nc(S)sc1CC(=O)NCC1(NC(=O)CC2(O)CCOC2)CCOCC1 c1(C(N(C2CCCCC2NC(C2CCOCC2)=O)C)=O)ccc2nc(O)oc2c1 N1(C(=O)CN2C(=O)CNC2=O)CCC2(CCN(C(=O)CCCC(F)(F)F)C2)C1 C(CC(=O)NC1(C)CC(NC(C2CC(=O)OC2(C)C)=O)C1)(C(N)=O)NC(C)=O c1(CC(=O)NCC(CC)(C)NC(C2NC(=O)OC2C)=O)ccc(Cl)nc1 C1(C(=O)NC(c2cccnc2)C)(NC(C2C(C)=CCS2)=O)CCCC1C c1(C(=O)NCC2C(NC(c3c(C)nc(C)[nH]3)=O)COC2)cncc([N+](=O)[O-])c1 C1(CNC(C(C)(C)NC(N)=O)=O)CC2(CC2)CN1C(=O)C(C1CCCCC1)O C1(NC(CSCC=C)=O)CCCN(C(=O)CCN(CCCCC)C)CCC1 C(=O)(CC(C)(C)CC(F)(F)F)N1C(C(C)NC(=O)CCc2cncs2)CCC1 C1(C(=O)NCCn2cncn2)CCN(C(=O)Cc2c[nH]ccc2=O)C12CCC2 C1(NC(C(CC#C)N(C)C)=O)CCN(C(=O)C(C)(C)C(F)F)CC1C c1(CC)ncc(Cl)c(C(=O)NC(C)CC(C)NC(c2[nH]cnc2C)=O)n1 C1(C(=O)NC2CCCCN(C(CCC(=O)NC)=O)C2)CCc2c(n[nH]c2C)C1 c1(C(N2CCC(CCNC(=O)C=CC=C(Cl)Cl)C2)=O)cc2cccnc2s1 C=CCCC(F)(F)C(=O)N(CCCCN(C(=O)CNS(=O)(=O)CC)C)C C1(CNC(=O)CC2(C(F)F)CC2)C2CN(C(c3cscn3)=O)CC12 N1(C(C=CCC)=O)CCC(CC(C)NC(c2cnc(N3CCOCC3)s2)=O)CC1 Cc1csc(C(c2nnnn2C2CC2)NCCc2ncccn2)n1 N1(C(CCCC(CC)NC(CC(C)(CO)OC)=O)=O)CCC2(CNC(=O)N2)C1 C1(CC=C)(C(N2CCOC(C(C)C)C2)=O)CCCN1C(=O)C(C)NC(N)=O c1(NC(C(=O)Nc2cc(C(C)(C)C)ncc2)=O)ccc2c(c1)C(=O)CC2 N1(C(c2cccc(OC)n2)=O)CC2CC(NC(c3ccncc3C)=O)CC1C2 Cc1ccc(C)c(C(C)NCc2ccccc2Sc2cnc(CC(C)C)s2)c1 c1(C(N2C(COC)CN(C(=O)CN(C)C(C)C)CC2)=O)cc2cccnn2n1 C1(C(=O)NCC2(CNC(C(COCC)(C)C)=O)CC2(F)F)CC2(C1)CC21CC1 Cc1c(NC(=O)C(C2CCN(c3ncc(C(F)(F)F)cn3)CC2)C)ccnc1Br c1(C(N2C(C(CNC(CC(C)O)=O)(C)C)CCC2)=O)cccn2ccnc12 N1(C(C(CC)C)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1C c1(C(N(C2CCN(C(C3CC4(CC4)C3)=O)C2)C)=O)cc(O)ncc1Br CCC(C)(CNC(=O)C(Cc1ccccc1)OC)NC(c1coc(C(F)F)c1)=O c1(C(=O)Nc2ccc(OC)cc2Br)n[nH]c2c1CN(Cc1cnn(C)c1C)CC2 C(C(O)CC(F)(F)F)NC(C1CCCN(Cc2cn(CCOC)nn2)C1)=O N1(C(CC(CC)(F)F)=O)CC2CC(NC(=O)CSc3ccncc3)CC(C2)C1 CC(CC(=O)N(C)CC1CCCN1C(=O)CCOC1CCC1)C(F)(F)F Cc1ccccc1NC(=O)CN(C(=O)Cc1ccoc1)C C1(C(=O)NC(C)CC2CCCCC2)CCN(C(C2CC(F)CN2C)=O)C(C)(C)C1 Cc1cccn2c(C(N3CCC(C)(CCNC(=O)C(C)O)C3)=O)cnc12 C1(NC(c2n(C(C)C)ncc2Cl)=O)CN(C(=O)C=C(Cl)Cl)C2(CCC2)C1 c1(OC(C(c2ccccc2)N(C2CCCCC2)C)=O)ccc[n+]([O-])c1 CCC(CC)C(=O)N(CCN(C(=O)CC1CC1(Cl)Cl)C)C(C)C O1N=Cc2ccc(cc2)NC(=O)C1.C(=O)(C(O)C1CCCC1)N(C)C N1(C(c2nnn(CC)c2C)=O)CC2CC(NC(c3ccc(C(C)C)o3)=O)C(C2)C1 C1(NC(c2ccc(CC)s2)=O)CCC(N(C)C(C2(CC(F)F)CCC2)=O)CC1 C12(NCCCCCC(N)=O)CCC(n3cc(C4CC4)nn3)C1C2 CCCCS(=O)(=O)CC(=O)N1CCOC(CCNC(=O)C(C)CN(C)C)C1 N1(C(C(CC)NC(N)=O)=O)C(CNC(=O)CCc2ccncc2)CC2COCC12 C=CC1CN(C(=O)C(F)C2CC(NC(=O)C#CC(C)C)C2)CCO1 C(O)(CCN=c1[nH]nc(C(F)(F)F)o1)(C(F)(F)F)c1scc(C)n1 C(N=C(NCc1cccs1)NCC1CCCOC1)c1nnn(C)n1 c1(C(=O)NC2CN(C(c3nc(OCC)sn3)=O)CC2F)cc2c(cn1)COCC2 N1(C(Cn2c(C)ccn2)=O)CC2CC1CN2C(=O)C(C)(O)c1ccccc1 n1(C(C)C)cccc1C(=O)N(CC(C)N(C(=O)C=CC1CCOC1)C)C CC(C)(C)C(CNC(=O)C(O)c1ccco1)C(=O)NC1CCCCCCC1 N1(C(CCc2cccc(OCC)c2)=O)CC2CCC(N)CC2C1 N1(C(CSCCC)=O)CC(NC(C2(COCC)CC2)=O)C(c2cnn(C)c2)C1.C(C)(C)N c1(C(N(C2CCN(C(=O)CC3CC=CCC3)C2)CC)=O)ccccc1OC N1(C(C(C)C2CCCC2)=O)CC(CNC(=O)CC(=O)NC2CC2)CC1(C)C CCCC(C)(CCC)C(=O)NCC1CN(C(=O)C2=C(Cl)CCC2)CCC1(C)C N1(c2cccc(C)c2)C(=O)COC(NC(=O)COc2cn(C)c(C(N)=O)n2)C1C C1(CC)CCCCC1NC(C1(CO)CN(C(=O)COC(C)=O)C1)=O.C(C(C)(C)C)O CC1CN(CCCS(=O)(=O)N2CCOCC2)Cc2c[nH]nc21 O=C(N=c1[nH]oc2ncccc12)CC(N1CCCC(n2nc(Cl)ccc2=O)C1)=O Cc1cccc(F)c1CC(=O)NC1CC(CNC(C2CCC(C)CC2)=O)C1(C)C N1(C(C(CCCOC)C)=O)CC2CCC(C1)N2C(C1CCC1c1nc[nH]n1)=O C(=O)(C(CNC(C1(NC2CCC2CC)CC1)=O)C(C)(C)C)N(C(C)C(F)F)C C12(NC(c3c(C)cco3)=O)CCCCC1CN(C(c1nc(O)nc(O)c1N)=O)C2 C1(C(N2CC(CNC(C(CC)C3CCC(=O)N3)=O)C2)=O)CCCN(C(N)=O)C1 c1(N2CC(C)C(NC(c3cc(C(F)(F)F)n[nH]3)=O)C2)ncccc1S(C)(=O)=O CC(C)CCCCCC(=O)NCCC(N1CCC(N=[N+]=[N-])C1)=O CC1(C)CC1(C(N1CCC(CC(N)=O)C1)=O)NC(=O)Cc1ccsc1 C1(NC(c2c(CC)scc2)=O)C(CNC(=O)CO)CCC12CCC2 CCC(CC)C(=O)N1CCC(C(C)C(=O)NCCC(F)F)C1 C12CCCC(C1)N2.CC(C(=O)NCC(C)N(C)C(c1ccsc1)=O)NC(N)=O N1(C(c2nn(CC)c(O)c2)=O)CC(CO)C2(C1)CN(C(c1cc(Cl)cnn1)=O)C2 c1(C(N2CCCC(CN(C(=O)C3=CCCO3)C)C2)=O)ccc(N)c(F)c1 N1(C(=O)Cc2ccccc2)CCCCCCC1C(N1CC(F)(F)C1)=O C1(NC(c2nncc(CCC)c2)=O)CC(CNC(=O)Cc2cnoc2)C12CCC2 c1(C(=O)NCC2N(C(CCC(C)C)=O)C3C(C2)COC3)ccc2nnn(O)c2c1 c1(C(N2C(C3CCCN(C(=O)C(F)F)C3)CCCC2)=O)ccc([N+](=O)[O-])cc1Br Cc1ccccc1OCC(N1CCC(CNC(c2cn(CC3CC3)nn2)=O)C1)=O c1(CCC(=O)N(C(C)C)CCNC(=O)CCC(N)=O)nnc(S)nc1O C1(NC(=O)Cn2cccnc2=O)CC12CCN(C(=O)C(F)C1CCC1)CC2 C12(C(N3CCC(CNC(C(C4CCC4)OC)=O)CC3)=O)CC1COC2(C)C Cc1cc(CN(C(=O)CN(C(=O)C(C)C#N)C)C)n(C)n1 N#Cc1cc(Cl)c(C(N2CCC2Cn2cc(C3CCCOC3)nn2)=O)s1 c1(N(C(c2ccc(CNC(CCC3C(C)C3)=O)o2)=O)CCO)cc(C)cc(C)c1 C1(NC(c2cc(CC)c(CC)o2)=O)CCN(C(c2cccnc2NC)=O)CC1F CCCC(C)CC(C(=O)NCCCF)N1CC(C(=O)OCC)C2(CCCC2)C1 C12(CNC(c3ccn(C)n3)=O)CCCC1CN(C(C13CC1COC31COC1)=O)C2 C=CC(CCC)CC(=O)N1CC=CC1CNC(c1ccc(C(F)(F)F)s1)=O C1(CC(=O)NC2C(NC(C(CC)NC(N)=O)=O)CCCC2)CCC(F)(F)CC1 c1(C(=O)OCC)cn(CC(=O)NCC(O)CN)nc1C(F)F.C(C(C)(C)C)=C c1(C(N(C2CCN(C(=O)C(C)(C)n3cncn3)CC2)CC)=O)[nH]ccc(=O)c1C Cn1cc(C=C(F)C(=O)NC(C)(C)CCNC(c2cc(C(N)=O)co2)=O)nn1 C(CCCC(CO)NC(C12CC(C)C1C2)=O)NC(c1c(Br)cn(CC)n1)=O C(CN=C(NCCCc1ccccc1)NCC12CCCCC1C2)C1(C)CCC1 N1(C(c2cc(CC)on2)C(=O)NCC)CCOCC1(C)c1ccccc1 C1(C(=O)NC(c2cnn[nH]2)C)CC12CCN(C(c1cncnc1)=O)CC2 c1(C(=O)OC)ccc2ccccc2c1NC(c1cc2ccccn2n1)=O c1(OC)cc(C(N2CCOC(CCCNC(=O)CCc3cnn[nH]3)C2)=O)n(C)n1 N1(C(CCC(C)N(C)C)=O)CCN(C(C23COC(CF)(C2)C3)=O)CC1C C1(=O)C2=NOC(C2)CN1.C1(C(N2CC(O)(C(C)C)C2)=O)CC(=O)CCO1 C(=O)(CCCCC(C)C)N1CCC(CNC(c2cccc(OC)c2F)=O)(OC)C1 C=C1CC2(C1)CC(C(=O)NCC1CCCN(C(C3(C4CCC4)CCC3)=O)C1)C2 c1(N2C3(CNC(c4c(C)noc4)=O)CCC2CC3)ncc2ncn(C)c2n1 C12(C(=O)NC(C(=O)OC)CSC)COCC1CN(C(c1ccncc1)=O)C2 C1(C2CCN(C(=O)COC3CCOC3)CC2)(NC(C2(C)C(C)(C)CCC2)=O)CC1 N1(C(c2c(C)cccc2Cl)=O)CCC2(CCCC2NC(=O)C(C)C2CC2)CC1 N1(C(C#C)C)CCN(C(=O)CC2(C(=O)NC3CN(C(=O)NCC)C3)CCC2)CC1 C(c1cccc(C#N)c1)=CC(=O)NCC(C(C)C)(C)NC(=O)CC(C)F Cc1ccc(Cl)c(C(=O)NC2CC(F)CN(C(=O)C(C)(C)N(S(C)(=O)=O)C)C2)c1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCN(C(C(CC(C)C)C)=O)C(C)C O=C(C1CCCc2sccc21)NCC1CC(NC(C2CCCC23OCCO3)=O)C1 C(=O)(CC(C)C(F)(F)F)NCC1N(C(C2CCN(C(N)=O)CC2)=O)CCC(C)C1 CN1CC(=O)N(CC(N2CC(NC(c3cc(Cl)sc3Cl)=O)CC(O)C2)=O)C1=O c1(NC(C(N2CCC(N(CC)CC)C2)c2cnc(Br)s2)=O)ccc(F)cc1 C12(CNC(c3c(CC)n(CC)nn3)=O)CN(C(C3CCCCS3)=O)CC(F)(C1)C2 CCC(CC(=O)NC(C1(O)CN(C(=O)C(F)(F)C2(O)CCCC2)C1)C)C1CC1 C(CC)(C(O)C(C)C)CONC(C1(C#C)CN(C(=O)CCC(C)CN(C)C)C1)=O CC(C)CCC(O)C(=O)NCc1cc(NC(=O)CN(C)C)cn1C.C1CCNS1.N CC1CC(C(=O)N(CC(O)CN(C)C(c2nccs2)C)C)CCC1=O c1(C(N2C(C(=O)NCc3cc(OC)no3)CC=CC2)=O)cc(=O)n(C)cn1 N1(C(C(=Cc2ccc(F)cc2)C)=O)CCCN(C(C2CCSC2)=O)CCC1 C(=O)(CCN1CCCO1)N1CCC(NCc2cn(C)nc2)CC1 C1(NC(C=CC)=O)CCCCC1NC(c1ccc(CN(C)C)cc1)=O C=CC(C)(C)C(=O)N1CCC(C(N2CCS(=O)CC2C)=O)O1 N#Cc1cn(CC(N2CCN(C(=O)CNC=O)CC(CO)C2)=O)c(=O)nc1O c1(NC)cc(OC)cc(OC)c1SC.C1(c2ccccc2)CC(=O)N1 C(CCC1CCC1)(C(=O)N1CC2C=CC2C1)NC(C(c1ccn(C)c1)C)=O c1(C(=O)NCC(C)NC(C2(F)CCCCC2)=O)coc2ccc(O)cc12 c1(NCC2N(S(CC(C)C)(=O)=O)CCCC2)ncnc2c1cnn2C CC(CNC(C1CC(C)(C)CO1)=O)CC(=O)NCC(C)Cc1cn[nH]c1 C1(NC(COCCOC)=O)CCCC1NC(=O)C(C)Oc1cccnc1 C(c1ccc(F)c(F)c1)=CC(N1C(CC)C(NC(C2CC(OC)C2)=O)CC1)=O CCC(C)C(C)CNC(C1(NC(=O)Cc2ncoc2C)CCCCC1)=O c1(-c2occ(C(=O)NCC3CCC(NC(C(C)C)=O)C3)n2)ccccc1Cl N1(C(C2N(CC)CCC2)=O)Cc2occ(C(=O)NC(C)(C)CC3CCOC3)c2C1 C1(NC(C2C(CCC)CCC2)=O)CN(C(=O)CCc2nnc(C)o2)CC12CCC2 C(=O)(CC(CNC(=O)C1=CCCC1)C1CCC1)NCCNC(C(C)(C)C)=O Cc1ccc(Br)cc1CCC(=O)NC(C)(CNC(C1C(C)C1C)=O)CO c1(C(N2C(C)CN(C(=O)COC(F)F)CC2)=O)cc(F)cc2nc(S)[nH]c12 C1(NC(c2[nH]nc3ccccc23)=O)CN(C(C2CCC=CO2)=O)CC2(CC2)C1 C1(C(N(CCNC(c2csc(-c3ccco3)n2)=O)CC)=O)Cc2cccnc2C1 C(=O)(C1=C(Cl)CCOC1)N(CC)CC1CCCN(C(=O)CS(N)(=O)=O)C1 c1(C(N2CC(C)CC(OC)C2)=O)cc2c(cc1N)OCCO2 Cc1ccc(COCC(=O)NCCC2(NC(=O)CC3CNC(=O)O3)CC2)cc1 C1(NC(=O)C=CC2CC2)CC2CCC(C1)N2C(c1n[nH]cc1I)=O Cc1cc2c(cnn2C)c(N(C)Cc2ccc(C(F)(F)C(F)(F)F)cn2)n1 Cc1cc(Cl)ccc1C(=O)NCC1(CNC(c2cn(C)nc2C(F)F)=O)CCC1 N1(C(CNC(CN(C)C)=O)=O)CCC(C2CC2)C1C(=O)NCC1(C)CCC(=O)N1 c12nc(C)c(c(C)c1Cl)NC(=O)NC2.C1(C(=O)NCC)CC12CC2(F)F.C(COCC)O c1(C(=O)NC2C(NC(c3ccc(CC)nc3)=O)CCC2)nn(C)c2c1COCC2 CC(CCNC(C1CCOC1)=O)NC(C1CC(CNC(=O)OC(C)(C)C)C1)=O c1(COC(=O)CCSc2ccc(Br)cc2)cc2cc(Br)ccc2o1 N1(C(C2CCC(CNC(CNC(=O)OC)=O)C2)=O)CCC2(CCC2)C(O)C1 N#Cc1cncc(C(N2CCCCC(C(=O)NC(C3CC3)C3CC3)C2)=O)c1 C=C(C)CCCC(=O)N1CC2CC(NC(c3cccn(O)c3=O)=O)C2C1 N1(C(c2ccc(C(=O)OC)cc2)=O)CCN(C(C2CNC(=O)N2)=O)CC1C(F)F C1(NC(C=CC(=O)N(C)C)=O)CCN(C(=O)CCC2CC(C)(C)CO2)C12CCC2 c1(N2CCCC(C)(COC)C2)nc(C)cc(=NC(C)c2ccc(C)c(C)c2)[nH]1 c12sccc1CC1CC(C1)CCNC2=O.C(=O)(C(C1CCCO1)C1CC1)N.CO C1(NC(CC(CNC(=O)Cc2cc[nH]n2)OC)=O)CCCC(F)(F)C1 C1(C(C)NC(c2cc(CC(C)C)on2)=O)CN(C(C2CCCOC2)=O)CCO1 C1(NC(=O)C=Cc2ccsc2)CCCN(C(c2ccn(C3CC3(F)F)n2)=O)CC1 C(=O)(C(=O)C(C)(C)C)N1CC2C(CNC(C3C(C=C)C3)=O)C2C1 c1(C(=O)NCC2CCN(C(=O)CC3CC4(CCC4)C3)C2)cc(Cl)c(F)cc1F C1(C(=O)NCc2csnn2)CCN(C(=O)c2cccs2)O1 c1(NC(C)=O)cnc(C)c(C(=O)NC2C=CCN(C(c3ccc(F)o3)=O)C2)c1 N1(C(COC2CCC(C)O2)=O)CCCC2CN(C(CCCCCC)=O)CC12 C12C3CN(CC13)C2=O.C1(O)(C(=O)NCC2(n3cc(Br)cn3)CC2)CCSCC1 CCC(CC)C(C)C(=O)NC(C(=O)N(C)CCN(CC)CC)C(C)C n1(CC)nc(C(=O)NCCC2CCCN2C(=O)C=CC2CCOCC2)c(C)n1 c1(NC(=O)OC(C)(C)C)ccc(C(N2CCC2c2cccs2)=O)cc1.N1(C)CCCC1 c1(C(=O)NC2CC3N(C(C(C)(O)C(F)(F)F)=O)C(CC3)C2)cc2[nH]ccc2cc1Cl c12ccc(cc1)CN1CCN(CC1)c1ccc-2s1.c1(C(CO)SC)ccccc1 c1(C(=O)NCC(C)C(=O)NC2CC(CO)C2(C)C)cccc(O)c1F Cc1nn(CCO)cc1C(c1nnnn1C1CC1)NCC(C)F C1(CC)(NC(c2cc(N(C)C)ccn2)=O)CCCN(C(c2cccn2C)=O)C1 C(=O)(CCC(C)(C)C)N1C(C)C(NC(=O)C(C)(C)c2ccno2)CC1 C(CC(O)C(=O)NCC1(O)CN(C)C1)NC(C(CC)n1ccnc1)=O c1(C(=O)NCC2(O)CN(C(C(C)SCCCC)=O)C2)cc2c(ccn2C)s1 c1(N2CCCC(Cn3ccnc3)C2)nc(N2CCOC(CF)C2)nc2c1CCC2 C1(C2CCN(C)CC2)(C(N2CC(NC(C3N(C)C(=O)OC3)=O)C(F)C2)=O)CC1 CS(=O)(=O)c1ccc(C(=O)NC2CC3CC2CC3O)c(N)c1 C(=O)(CC(F)(F)Cl)NCC1CCC(NC(C2(CC=C)COC2)=O)C1 C1(CCNC(Cn2c(C)ccn2)=O)CCCCN1C(=O)CC1CCNC(=O)C1 c1(CCCC(=O)NCCCC(C)NC(=O)CCC2CCC(=O)N2)ccc(F)cc1 C1(NC(C2CC3(CCC3)C2)=O)CCCC12CN(C(c1ccco1)=O)C2 C1(CNC(=O)CC2CCCN2C(C2CN(C(N)=O)C2)=O)CC12CCCCC2 N1(C(C(OC)OC)=O)CCC(C)(NC(c2cnn(-c3cccc(F)c3)c2N)=O)C1 N1(C(CCN(C(=O)C2=C(C)OCC2)CCS(N)(=O)=O)=O)CCC2(CCC2)C(NC)C1.CO c1(OCCC(C)C)cccnc1C(=O)NCC(C)CN(C)C(c1cnc(S)[nH]1)=O c1(OC)cc(OC)c(C(N2CCC2CNC(=O)C=Cc2ccccc2C)=O)c(N)c1 c1(N(C)C)cccc(-c2cn(CC(=O)NCCC3(C)COC3)nn2)c1 CCCC(O)CC(=O)N1CCN(C(c2ncc(Br)cc2C)=O)C(C)C1 c1(C(=O)NCCC2(O)CCN(C(C3(C=C)CC3)=O)C2)n[nH]c2c1CCCC2 N1(C(c2c(C)ccc(C)n2)=O)CCN(C(=O)CNC(=O)CC(F)(F)F)CC(O)C1 c1(C(N2CCOCC2C2CCCNC2)=O)cccc2[nH]c(-c3ccco3)nc12 C(CN=[N+]=[N-])(C(=O)N(C)Cc1c(C)cnn1C)NC(C(C=CC)O)=O C1(C(N(C(CC(CC)C)C)C)=O)CCN(C(=O)C#CC(C)(C)C)CC1(C)C N1(C(CCC(C)C)=O)CC2CCCN(C(C3CCN(C4CC4)C3=O)=O)C2C1 N12CC3(CO)CC1(C3)C2=O.N1(C2ON=C(CC)C2)CC(CC)CC(C)C1 C#Cc1ccc(CC(=O)N(CCC(C(C)C)NC(C2CCC3(CC3)C2)=O)C)cc1 c1(CC(N2C(C)(C)CC(c3cn(C4CCOC4)nn3)C2)=O)cc(F)c(F)cc1F C1(NC(c2c(CC)c[nH]c2)=O)CCCCC1NC(=O)C(C)CC1CCCCC1 Cc1c(F)ccc(NC(CNC(=O)OC(C)(C)C)CCS(C)(=O)=O)c1N.C C(N=c1cc(C(F)F)nc[nH]1)C1C(C(CNC(C(C(C)(C)O)F)=O)=O)CCC1 N1(C(C(C=CCCC)O)=O)CCN(C(c2ncccc2N)=O)CC1C(CC)CC C(CS(=O)c1ccccc1F)N1C(=O)NC(C)(C)C1=O C1(NC(C=C(C)Cl)=O)CCN(C(=O)CSCC2CCCCO2)C1C N1(C(C2(OC)CCOC2)=O)CCC(C2(O)CN(C(c3cncs3)=O)C2)CC1 N1(C(C(CC=C)C)=O)CC(C2CCN(C(c3ccc4c(c3)CNC4=O)=O)CC2)C1 C(C)(C(=O)N1CC2(CC2)CC1C)(C(C)C)NC(C=CCOCCOC)=O C=CC(O)C(=O)NCC1CC(OCC)C1.C12(CC(CO)C1)C(=O)N2 C12(C(N(CCC(C)NC(c3noc(C)c3Br)=O)C)=O)CCCN(CC1)C2 C1(NC(N2CCn3nccc3C2)=O)COC2(CCN(c3ncccn3)CC2)C1 C1(C(N(CC(C)NC(C(CC)NC(N)=O)=O)C)=O)CC(F)(F)CCC1(C)C N1(C(Cc2scc(C)c2)=O)CCC2CCN(C(C3(CCN(C)C)CC3)=O)CC12 c1(CC(=O)NCc2c(C(=O)NC(COC)CO)occ2)ncccc1F N1(C(CC(=O)N(C)C(C)=O)=O)CCCC2CN(C(C34CC(C)(C3)OC4C)=O)CC12 N1(C(c2c(C)ncs2)=O)CCN(C(C2CCc3c(ncn3C)C2)=O)C2(CCC2)C1 C(=O)(C1=CCCCCC1)N1CCC(N(C(Cc2ccc(C)nc2Cl)=O)C)CC1 c1(Cn2cc(-c3cc(C)sc3)nn2)nnc(N2CCCC2C2CC2)n1C C(=O)(C(CC(C)CCC)N1CCOC(CF)C1)NC(CC)(C)C C1(C(=O)NCC2C=CCN2C(c2cc(C(N)=O)no2)=O)CCCCCC1 Cn1ccc(C(=O)NC(c2cccnc2)C(=O)NCC(O)C2(Cl)CC2)n1 c1(OCC(=O)NC2CC(CCNC(=O)CC(C)C3CCCO3)C2)ccccc1F C1(CC#N)CN(Cc2cc[nH]c2)CCN1C(c1cc(C(F)(F)F)cc(Cl)c1)=O C1(C(N2CC3(CN(C(c4c(C(N)=O)cccc4)=O)C3)C2)=O)CCc2nn[nH]c2C1 C1(CNC(=O)NCC(C)O)COCCO1 C(CC(=O)Nc1csc(Cl)c1)(C(F)(F)F)NC(Cc1cn(CC)nn1)=O Cc1noc(CCC(=O)NCCOCCN(C(=O)CC2COC(=O)C2)C)n1 c1(OC)ccc(C(=O)C(=O)NCC2CCC(NC(=O)CCn3cncn3)C2)cc1 c1(C(=O)NCC2CC(C)N(C(c3scnc3Cl)=O)C2)cncc2[nH]ccc12 N1(C(C2(CO)CCN(C(Cc3ccc(C)nc3)=O)C2)=O)CCC2(CNC(=O)C2)C1 C1(C(=O)NCC(N(C(CSC(C)C)=O)C)C2CC2)CCCN1C1CCCC1 N1(C(CC(C)C2CC2)=O)CC2CC(NC(=O)CSCc3cccs3)CC1C2 c1(C2C(C(=O)NC3CC3C(=O)NCc3ccoc3)C2)ccc2ccccc2c1 c1(OC)ccc([N+](=O)[O-])cc1C(N1CC=CC1C(N1CC2CCCCC2C1)=O)=O C(=O)(C(CC(C)C)NC(=O)C(F)(F)F)NC(C)CNC(c1nc(C)n(C)n1)=O c1(C(=O)NC(C(C)(C)NC(COCCCCC)=O)C)oc(C2CC2)nc1C C(=O)(C(O)CCSC)N(C(C)CNC(c1cc(Cl)n[nH]1)=O)CC C=CC(C)(C)C(=O)NC1CCCN(Cc2cccc(Cl)c2)C1.C12CC1NC2=O O=C(CCS(=O)(=O)N1CCCCC1)NC12CC(NC(C3CC(O)C3)=O)(C1)C2 c1(CC(=O)NC2C(CCCc3cccc(C)c3)C2)cc(C)ccc1OC(C)C c1(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCSC)cccc(C(C)(F)F)n1 C1(C(=O)NC2CC(F)(CNC(=O)Cc3cnn(C)c3)C2)(CC)CCOCC1 N1(C(c2cccc(C)n2)=O)CCC(NC(=O)CC2OCCC2(C)C)C(O)C1 c1(OCC)ncc(C2=CCSCC2)o1 C1(C(=O)NOC2CCCCC2)(CC=C)CCCN1C(c1ccc(CO)cc1)=O C1(C)(C(N2C(C#C)CCC2)=O)CC(O)CN1C(C1CC1OC(C)=O)=O N1(C(CCOCCOCC)=O)CC2CCC2(CNC(=O)Cc2sccc2Cl)C1 Cc1cccc(Cl)c1C(N1CCCC1CN(C)C(c1cnn(C(C)C)c1C)=O)=O S(=O)(=O)(c1cnn(CC(F)F)c1)N(c1cncc(Br)c1)Cc1c(C)noc1 S(=O)(=O)(c1cccs1)CC(=O)NC(CC=C)CNC(=O)CC1OCCC1C CCC(C)(C#N)C(=O)NCCCOCCNC(=O)C(C)(C)C1CCOC1 CC1=C(C)CN(C(=O)CCC2CCCC(NC(=O)CSCC(F)F)C2)CC1 C1(C(C)C)(C(=O)NC(C)Cn2cncn2)CCCN1C(C12CSCC1C2)=O CCC(C)C(CC(=O)NCCC(=O)OCC)NC(=O)C(c1ccc(F)cc1)=O C(C(CC(C)C)NC(=O)Cc1csc(C)c1)NC(C(CN(CC)CC)F)=O CC1(NC(=O)CC2CC(C)(C)CO2)CCCN(C(=O)Cc2csc(S)n2)C1 Cc1nccc(C(=O)N(C)CC2CCCCN2C(=O)C(C)NC(N)=O)c1N c1(C(=O)NCC(CO)NC(CC=C)=O)ccc(N2CC=CC2)cc1 C1(NC(C2(OC)CC2)=O)CCC2CC1CN2C(=O)CC1(CO)CCCC1 N1(C(C(C)C)=O)CCN(C2CCCN(C(=O)C=C(Cl)Cl)C2)CC1.C(C=O)SCC c1(C(=O)NCCN(C(=O)Cc2c[nH]nc2C)CC)cnn2c1OCC(OC)C2 C1(NC(CC(=C)C)=O)CN(C(C2CSCN2C(=O)OC(C)(C)C)=O)C(C)(C)C1 CC(C)C1=NOC(C(=O)NCC(c2ccc(C#N)cc2)O)C1 CCCCC(C(=O)N(CC(C)C(F)(F)F)C)NC(=O)CN1CCCCC1C c1(C(N(CCCNC(C2CCC2C(F)(F)F)=O)C)=O)cccc(Cl)c1O N1(C(CC2CC(=C)C2)=O)CCC(CNC(c2csc(C(N)=O)n2)=O)(OC)C1 N1(C(CNC(=O)OC)=O)CCN(C)C(CNC(C23CC2CN(C(C)=O)C3)=O)C1 N1(C(c2ccc(C)cc2N)=O)CC=C(C(C)(C)C(=O)N2Cc3cccnc3C2)C1 C=C(C)CC(C(=O)N1CCC(O)(CC)C1)NC(C1CC(O)C(F)C1)=O c1(C(=O)NCC2CCC(NC(CC(C)C(F)(F)F)=O)C2)noc2c1CCCCC2 c1(NC(C2SCCN(C(c3c(C)cnnc3)=O)C2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] CCC(C)CC(=O)C(=O)NC1CCC(CCC(N2CCNC(=O)C2C)=O)C1 N1(C(C(C)OCC=C)=O)CC(CCC)(NC(=O)CNC(=O)C)C1 c1(NC(=O)NC(CC)C2CC2)cc(CNC(=O)OC(C)(C)C)ccc1O c12c3ccc3c1[nH]c2=O.N1(C(C2(COC)COC2)=O)CCC(OC)C1.OC.OC C(=O)(N=c1cc(C2CCCCC2)[nH][nH]1)C1N(C(Cn2c(C)cc(C)n2)=O)CCC1 c1(C(N2C3CC(CNC(C(CCCC)C)=O)(OC3)C2)=O)cc2c(C)cccc2o1 C1(NC(c2cnc(OCC)nc2)=O)CC12CCN(Cc1ccncc1O)CC2 c1(C(=O)NCC2N(C(C(c3cccs3)OCC)=O)CC2)ccnn1C C1(C2(O)CCN(C(C3CC3F)=O)CC2)(NC(C(C(C)C)NC=O)=O)CC1 N1(C(C2C=CCC2)=O)CCN(C(=O)C=Cc2cn[nH]c2)C(c2ccccc2Cl)C1 c1(C(N2CCN(C(CS(=O)(=O)NC)=O)C(C)C2)=O)cc(F)c(F)c(O)c1F C(=O)(C(C)(C)CC(=O)N1CCC(C(=O)Nc2cnn(C(F)F)c2)C1)OC C=C(Cl)CCC(=O)NC(c1cccnc1)C(C1CCOC1)NC(C1(C)CCCCC1)=O c1(C(C(C)CC)=O)ccc(C(C)C(N2CCCC(NC)C2)=O)cc1 c1(OC)cc(C(=O)N(C2CN(C(C3CC(C)C3)=O)CCC2C)C)ccc1F c1(CC(=O)NCCC2CC(NC(C3CC4CC4C3)=O)C2)ccc(Cl)cn1 c1(C(N2C(C(C)NC(c3coc(Cl)n3)=O)CCC2)=O)c(F)cc(F)c(F)c1F C1(NC(C(C)CN(C)C(c2ocnc2C2CC2)=O)=O)CC2C(C1)C2(F)F N1(CCC)CCCCC1C(N1CCCC(CNC(=O)CC2CCN(C)CC2)C1)=O C(=O)(C1COc2ccccc21)N1CC(NC(C2C(C)(C)CCC2)=O)C(F)CC1 C1(C(=O)NCc2cc(COC)no2)CN(C(C2COCCN2C)=O)CCN1C N1(CCNCCNC(N(c2onc(CC)n2)C)=O)CCC(O)CC1 C1(NC(C(C(C)O)C)=O)CCCN(C(=O)C=Cc2cccc(F)c2)C1C C1(C(N2CC(NC(C3(C(=O)OC)CC3)=O)C2)=O)CCc2nc(C)ncc2C1 C1(C(=O)NCC(CCCC)NC(=O)Cc2[nH]cnc2C)COC2(CCC2)C1 C(=O)(CC(CC(C)C)NC(C1CC(C)CC(=O)N1)=O)NCCCOC N1(C(C=Cc2c(C)ccnc2)=O)C2CC1CN(C(=O)C(C)CCN(C)C)C2 c1(C(=O)NCC(=C2CN(C(C3CC=CCO3)=O)C2)F)c(Cl)nc2ccccn12 C(=O)(CCCN(C)N=O)NC(C)CC1CN(C(C2CCC(C)(O)CC2)=O)C1 CCCC(C(=O)NC1(C(N2CCOC(CF)C2)=O)CCCC1)NC(N)=O C=CCC(CC(C)C)C(=O)NCC1CN(C(=O)CC2CCCCC2)CC1O c1(C(=O)NCCC2(O)CN(C(C(CC)(C)C(N)=O)=O)C2)cc2cnc(Cl)cc2s1 c1(CC(=O)NC2CCN(CC3N(CC)CCC3)CC2)ccc([N+](=O)[O-])cc1 N1(C(c2ccc(CCCCC)o2)=O)CC(NC(=O)C(F)CC2CC2)C(N=[N+]=[N-])C1 C#Cc1ccc(C2CC2C(=O)NC2(CNC(=O)C(C)(C)C(=C)C)CCOC2)cc1 C1(C(C2CN(CC(=O)N(C3CCN(C(C(C)C)=O)C3)C)C2)=O)CCC(=O)N1C Cc1ccc(OCC(=O)NC(C)(CNC(=O)Cn2cc(CO)nn2)CO)c(F)c1 C(CCCCCNC(C1CCC1c1nc(S)n[nH]1)=O)NC(=O)C(Cl)=CCl c1(NC(=O)CCn2cccc2)c(C(F)F)nc2n1CCCC2 CS(=O)(=O)c1sccc1C(=O)NC1CC2(C1)CN(C(=O)Cc1cccnc1O)C2 C(=O)(CC(C)(C)C)NC(C(=O)NC(C1N(C(c2c(C)con2)=O)CCC1)C)C Cc1nc(C)c(CNC(=O)C(C2CCCC2)NC(c2cnn(C)c2N)=O)[nH]1 C1(NC(C(C)Cc2cnn(C)c2)=O)CN(C(=O)COC(C)(C)C)CC1(C)C C1(C)(CNC(C2C(CC)C2)=O)CCCN1C(c1cc(C)c[nH]1)=O C1(CNC(C(CC)(F)F)=O)CCCC2(CN(C(C3(CCOC)CCCC3)=O)C2)O1 C1(CC(=O)NC(CCOC)CNC(=O)C(C)C)CCS(=O)(=O)C1 c1(CNC(N2CC(c3cccnc3)CC(C)C2)=O)cc(Cl)c2c(c1)OCCO2 c1(CN(C(c2cc(N3CCCC3)ccc2O)=O)CC2C(C)C2)cccc(C#N)c1 c1(N2CC(CCC)N(C(=O)OC(C)(C)C)CC2)cncc2nnnn12 C1(CC(N2C3(CN(C(CC(=O)OC)=O)C3)CC2)=O)C(C)OCC(=O)N1CC C1(C(N2CCC(NC(CC3N(CC)CCC3)=O)CC2)=O)CC(C)(C)OC1(C)C C12(CC(NOCCOC)=O)CCC(NC(C3CCCC3OC)=O)(CC1)C2 CCC(C)(C)CC(=O)N1CCC(c2ccccc2)C(NC(=O)C(C)CF)C1 c1(C(=O)NCC2C(C)CCN(C(=O)CC3CCC(C)C3)C2)nc2ncccn2n1 c1(C(=O)NNC(=O)C2CC3CCC2C3)ccnc(F)c1Br C(CN=c1[nH]cncc1I)C1CCC(NC(c2cncc(OC)n2)=O)C1 c1(CCC(=O)NCCCCC(C)NC(=O)Cc2nnnn2C)ccc(F)c(F)c1 c1(OC)cccnc1C(=O)NC(CCN(C(=O)C(C)CO)C)c1cccs1 CCC(O)(CC)CC(C)(C)n1ccnc1-c1ccc(Cl)cc1 C#CCCC(c1nnnn1C1COC1)(NC1CCS(=O)CC1)C.C(CS(C)(=O)=O)N N1(C(C2CCCC2CNC(c2ncccc2F)=O)=O)CCn2ncc(O)c2C1 C(=O)(C1=CC(C)(C)C1)N(C1CCN(C(C2C(CC)CCO2)=O)C1)C CC(C)C(F)(CNC(=O)C=Cc1ccc[nH]1)C(=O)NCC12CC(CO)(CO1)C2 CCCS(=O)(=O)NC(C)C(=O)N(C1CCN(C(C2(F)CCC2)=O)C1)C CCC(C)(CNC(=O)Cn1ccnc1)C(=O)NCC(O)CC1CCC1 c1(OC)ccccc1C=CCNC(N1CCN(C2CCNCC2O)CC1)=O Cc1cc(C(N2CCCCC(NC(=O)COC3CCCC3)C2)=O)nc(O)n1 C=CC(C)(C)CC(=O)NC1CC(CNC(c2ccnc(C)c2)=O)C1(C)C Cc1noc(C)c1C=CC(=O)NCC=C1CCN(C(=O)CCC(C)N(C)C)CC1 C(=O)(C(CC(C)C)NC(c1cnn(-c2ccc(C)cc2-c2nn[nH]n2)c1)=O)OC c1(NCC2N(C(C(C)=C(CC)C)=O)CC=C2)ccc(C)c(C(=O)OC)c1 c1(C(=O)NCC2(C)CCC(NC(CN(CC)CC)=O)CC2)cc2n(c1)CCOC2 N1(C(CC=CC)=O)CC2C3CCC(C2C1)N(C(=O)Cc1csnc1OC)C3 CC(C)C(C(=O)NCC(C)(C)NC(=O)CCn1ccnn1)N(C)C C#Cc1cc(C(N2CC(CC=C)(NC(c3ccoc3Cl)=O)C2)=O)cc(F)c1 C=CCC(C)(C)CC(=O)N1CCC(O)C(NC(C2CC3(CSC3)C2)=O)C1 Cc1cc(Cl)ccc1C(=O)NCC(O)CNC(c1c(C)[nH][nH]c1=N)=O C(=O)(CCC(C)(F)F)NC1(CNC(c2ccc(C(=O)OC)s2)=O)CC1 C1(NC(c2c(C)con2)=O)CN(C(c2csc(CS(C)(=O)=O)n2)=O)CC12CC2 Cc1cc(C(N2C3CN(C(c4ccc(F)c(F)c4O)=O)CC23)=O)ccc1[N+](=O)[O-] c1(C(=O)NCC2C(CNC(c3c(CC)[nH]cc3)=O)C2)c(C(F)(F)F)cccc1C Cn1ccc(-c2cn(Cc3ccc(C(N4CCC4)=O)o3)nn2)n1 C(C(C)C)(C(O)C(=O)NCC1(F)CC(NC(C23CCCCC(F)(C2)C3)=O)C1)OC CCCCCCC(CC)C(=O)N1CCCCC1CNC(C1CC(=O)C1)=O CS(=O)(=O)CCC(=O)NCC1CN(C(=O)C=Cc2cncs2)C2CC12 c1(C(N2CCC3(CC(NC(CC(C)O)=O)C3)C2)=O)ccc2[nH]c(=N)n(C)c2c1 C#CCCC(=O)NCCCOCCCNC(=O)C(c1ccn(C)c1)C c1(C(=O)NCC2N(C(c3c(C)c[nH]n3)=O)CCC2)cc(C#N)c2n1CCCC2 C#Cc1cnn(C)c1C(=O)NCC1CCCC1C(=O)NC1CC1.N1(C)CCC(CC=C)C1.C=O CC(CO)(C(=O)NCC1CCN(C(=O)CCc2cncs2)C1)c1ccc(F)cc1 C(=O)(C(CCSC)NC(=O)CCCNC(c1cncc(Br)c1)=O)NC C1(CN(C)C(C2SCCS2)=O)CCCC(NC(=O)CN2CCCC2=O)C1 N1(C(N(C(CC)CO)CSc2ccccc2)=O)CCN(C2CCCCC2)C(C)C1 C(=O)(C1CCCc2c[nH]nc21)NC1CC(CNC(CN2CC(C)(C)C2)=O)C(O)C1 C=Cc1ccc(C(=O)N(CC(C)N(C)C(c2cc(CC(C)C)[nH]n2)=O)C)cc1 C(=O)(C(C)(C)CC(=O)NC1CC(CC(=O)N(CCCN(C)C)CC)C1)OCC C(c1c(F)cccc1F)=CC(N1CCC(CNC(c2c(C)cc(C)o2)=O)C1)=O N1(C(CC(C=C)(C)O)=O)C(CNC(=O)C(C)(C)F)CC2COCC12 Cc1ccc(C(=O)NCCC2(C(=O)NCC=CC(C)(C)C)CC2)c(F)c1 c1(C(=O)NCC23C(CN(C(CC4(OC)CC4)=O)C2)CC3)cc(C)n(C)c(=O)c1 C12(NC(CSCCCC)=O)CCCC(NC(=O)C(F)=C3CCCC3)(C1)C2 Cc1ccc(CC(=O)NC2CC(NC(=O)Cc3n[nH]c(C)n3)C(O)C2)cn1 Nc1cccc(C(=O)NC2(CCNC(=O)CC3CC3c3cccc(Cl)c3)CC2)c1 c1(CC(=O)N(CC(C)N(C(=O)CSCC(N)=O)C)C)ccc(-c2nc[nH]n2)cc1 Cc1c(N)ccc(C(N2CCC2CNC(C2CCCCC2(F)F)=O)=O)c1Cl C1(CCOC)(C(=O)NC(c2nccs2)C)CCN(C(=O)CC=C(Cl)Cl)CC1 N1(C(C=O)CC(C)C)CCC2(CCCN2S(=O)(=O)CC(C)C)CC1.C(=O)(CSC)OC C1(C(=O)NCC2C(CNC(c3cnc(O)s3)=O)C2)CCc2nc[nH]c2C1 C1(C(=O)NCC(C)CN(C)C(c2n[nH]cc2C2CC2)=O)CCS(=O)(=O)C1 CC1(CS(C)(=O)=O)CCN(C(c2ncc(C(=O)O)s2)=O)C1 Cc1cc(Br)ncc1C(C(=O)CCC(=O)N(C)C)=O.c1(N)ccc(C(=O)NC)cc1 C(CCC(F)(F)F)N(C(=O)C=CC1CCCN1C(c1cccc(F)c1)=O)C CC1(CC(=O)NC2CCCCC2NC(=O)Cc2ccccc2Cl)CCS(=O)(=O)N1 C(c1cc(Cl)c2c(c1)OCO2)=CC(N1CCC(CNC(c2cc(Cl)no2)=O)C1)=O c1(NC(CNC(c2ccccc2F)CCOC)=O)cccc2nnn(C)c12 c1(-c2c(C(c3nnnn3C3CCC3)NCC(=C)Br)c[nH]n2)ccc(Br)cc1 C1(CN(C(=O)C(N)=O)C)CN(C(c2[nH]cnc2C#N)=O)CCO1 c1(CNCCN2CCN(C(C=CC=CC)=O)CC2)c(F)ccc2occc12 Cc1c(C(N2CCC(CO)C2)=O)[nH]c2ccc(C(N3CCCC(F)C3)=O)cc12 C#Cc1ccnc(C(N2CCC(CCNC(=O)CSc3nncs3)CC2C)=O)c1 N1(C(CN(C)CC)=O)CC2CC(NC(=O)COc3ccc(Cl)c(Cl)c3)CC1C2 C=C(C)C(C)(C)C(=O)N1CCC(NC(=O)C(c2ccccc2OC)=O)C(CC)C1 c1(C(=O)NC2CCC(CNC(Cc3cccc(C)c3)=O)C2)sc2nccn2c1C c12cc([nH]n1)C(=O)N1CCC(C1)CNC(=O)C1(CC1)OC2.Cc1ccccc1 O(NC(=O)C(c1cccnc1)NC(C1CC1OC(C)=O)=O)C(C(=O)OC)(C)C N1(C(c2nc(CC)oc2)=O)CCC(CNC(=O)CCc2cc(C)cs2)C12CCC2 C1(N(C)C(C2CS(=O)(=O)C2)=O)CCCC(NC(c2cc(Br)n[nH]2)=O)C1 C1(C(=O)NCCN(C(=O)Cc2sccc2C)CCOC)OCCC1C N1(C(c2ncn(C(C)C)n2)=O)CCCC(CO)(NC(C2CCOC2)=O)C1 C=C(C)COCC(=O)NCC=CC(=O)NC1(C(C)C)CC1 N1(C(CCOC)=O)CCC2CCN(C(c3cc(C)cc(F)c3)=O)CC2C1 C1(NC(C=C(C)C)=O)CCN(C(=O)Cc2cc(C)cs2)CC1C(C)C C1(CNC(C(CCC)NC(N)=O)=O)CCC(F)(CSC)CC1.N12CCC1C2=O Cc1nn[nH]c1C(=O)NCC#CC(=O)NC1CC1(C)C(F)F c1(C(=O)NC(C2(CNC(C(C)c3cccs3)=O)CC2)C)ccnc(S(N)(=O)=O)c1 CC1CC2CN(C(=O)C(N3CCCC(c4ccc(Cl)cc4)C3)=O)CC2N1C1CC1 C1(NC(C(CC)c2ccccc2)=O)CCC(NC(=O)CCS(C)=O)CC1 C1(C2CC2)(CC(=O)N(C)Cc2ccn(C)n2)CC1.C12CC(C1)C(=O)NC2C n1(CC=C)cc(C(=O)NCC(C)N(C)C(c2cn(CC3CC3)nn2)=O)cn1 C#Cc1ccc(C(=O)OCC)cc1C.c1(O)ccccc1.C1(C)C(=O)N(C)CCO1 C(=O)(CCC(CF)CF)NCCC(C(=O)N(CCN1CCCC1)CC)O c1(SCC(=O)NCC(C)N(C(=O)CS(=O)(=O)N(C)C)C)ccsc1[N+](=O)[O-].C N1(C(C(CC)COC)=O)CC2=C(C1)CN(C(c1ncc(C)cc1OC)=O)C2 c1(CC(=O)NCCC2N(C(C(CC=C)C)=O)CC(F)(F)C2)ccc2sccc2c1 C(=O)(C(O)C(F)(F)F)NCC=CCNC(c1nnc(C)o1)=O N1(C(c2ccc(OCC)cc2)=O)CCC2(NC(c3ccc(=N)[nH]n3)=O)CC2C1 c1(OCC(O)CSCC2CCCC23CC3)ccc(Cl)cc1.N12CCN(CC1)C(=O)N2 c1(CC(N2C(CNC(CN(c3ccccc3)C)=O)C=CC2)=O)cccc(Br)c1 N1(C(C2CCN(C(C3C(COC)CC3)=O)C23CC3)=O)CCC(O)(C2CC2)CC1 c1(CNC(c2c(OC)scc2)=O)ccc(CNC(C2COCCO2)=O)c(F)c1 CC(C)C(C(=O)NC(c1ccsc1)C)NC(=O)C(=O)NC1CC1 n1(CC(=O)NCC=CCNC(C2CCC3CCC23)=O)nc(O)ccc1=O n1(C(CCN2CCCCC(NC)C2)C)cnc2ccccc12 CC1CC(NC(=O)CCc2nc(-c3cccs3)no2)CN1C(C1CCC=CO1)=O c1(-c2ccc(C(C)=O)cc2F)cc(C(=O)NCCC(C)(C)O)c2cn[nH]c2c1 N1(C(C2N(C(c3ccc(C#C)s3)=O)CC(O)C2)=O)CCC2(CCOCC2)C1 N1(C(C(CC)N(C)C)=O)CC2CCC1CN2C(c1cnn(C)c1Br)=O C1(NC(=O)CC23CCCC2C3)CCCCC12CCN(C(=O)CCCF)CC2 C1(C(=O)NCCC2(NC(C3C(C)C3)=O)CC2)CCC2(CCCC2)CC1 N1(C(C(C(C)F)(F)F)=O)CC2CCCC(C1)N2C(C1CC1(C)C(F)F)=O C1(C(=O)NC2(C)CCCN(C(CCc3ccn(C)n3)=O)C2)CCCCCC1(F)F C(=O)(C1=CC(O)C(O)C(O)C1)N1C2CC(CN(S(CCC(=O)OC)(=O)=O)C2)C1 CCC(C(=O)NC(C(=O)N1CC(C2CCCOC2)C1)C1(O)CCC1)OC C12C3CCC1CC(C3)C(=O)N2.C(=O)(C(=O)N(C)C)NC(C1CCO1)C c1(NC(=O)NC2(C(=O)O)CCOC2)ccc(OCC(F)(F)F)cc1 C1(NC(C2(CC)CCCN2C(=O)CC2COCC(C)O2)=O)CC2COCC(C1)C2 C(c1ccc(Cl)cc1F)=CC(=O)N(C1CCCN(Cc2cccc(C)n2)C1)CC C12(C(=O)NCC3C(NC(c4c(C)cc(C5(C)CC5)o4)=O)CCC3)CC(C)(C1)OC2C N1(C(C(F)OC)=O)CCC2CCN(C(=O)CSCc3ccccc3)CC12 Cc1cc(N(C(=O)CCC(C)NC(=O)CCC2CCC(=O)C2)C)cc(C)c1 c1(C(=O)NCC2CCCC(CNC(C3C(C=C)C3)=O)C2)cncc(C#N)c1 n1(CCC(=C)CO)cnc2c(N3CCC(CCCC#N)CC3)ncnc12 C1(C)(CNC(C2CN(C(CCC)C)C(=O)C2)=O)CN(C(=O)CC(=O)OC)CCO1 c1(C(=O)NCCCc2ccccc2Cl)cccc2c1[nH]c1ccccc21 N1(C(c2c(C)ccc(OC)n2)=O)CC2CCC1CC2NC(=O)C(F)=CC1CC1 c1(C(N2C(C(=O)OC)CC(O)C2)C(=O)NC(C)(C)C)cc(C)cc(Br)c1 c1(C(=O)NC2CCN(C(CC(C)F)=O)C23CCC3)cc2cnccc2cc1F N1(C(c2cn(C)cc2C(F)(F)F)=O)CC(NC(=O)C(=O)C2CC2)CC2(CC2)C1 c1(C(CNC(=O)CCCn2ccnn2)NC(C2CC23CCC3)=O)cccc(Cl)c1 C1(C)(CNC(CCOC)=O)COCCN(C(C)=O)C1.C12CC(C1)C(=O)N2 N1(C(c2cnc(C)s2)=O)CCC(NC(=O)C(F)(F)CC2CC2)CC1c1ccccc1 c1(CC(=O)NCCOC(CNC(CC2CCN(C)C2)=O)(C)C)ncc(F)cc1F C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NCCCN(C(C(CC)CC)=O)CC c1(C(=O)NCC(C)N(C(c2c(C)nc(C)[nH]2)=O)C)ccnc2ccc(O)cc12 C1(CNC(Cc2c(C)n[nH]c2C)=O)CCN(C(=O)CC(O)C2CC2)C1(C)C c1(-n2cc(CN(C(=O)CCC3CC3(C)C)C(C)C)nn2)cccnc1C(F)(F)F c1(OCC(=O)NC2CCN(C(COCC#C)=O)C2)cccc(C(N)=O)c1 C1(NC(C(c2cscn2)N(C)CCOC2CC2)=O)CCCSC1 c1(C(=O)NC2CCCN(C(CC3CN(C)C3)=O)CC2)ccc(F)c2ccsc12 c1(C(=O)NC(CNC(C(C=C)O)=O)CO)c(C(=O)NC)cnc2ccccc12 N1(S(C)(=O)=O)CCC(NC(C2CC3CC3N2C(=O)Cc2nc(Cl)cs2)=O)CC1 CCC(C)CC(C)C(=O)NCCC(=O)NCC(=O)NCCCN(CC)CC c1(C(=O)NC2(CNC(c3c(C)ccs3)=O)COC2)cc(Br)c(Cl)cc1F C1(NC(C=CCOC(C)(C)C)=O)COCCN(C(C2CC(Cl)(Cl)C2)=O)C1 C(C)(CC(F)(F)F)N(C(C1C(NC(CCCOC(C)C)=O)CCC1)=O)C N1(C(CCCC)=O)CCN(C(=O)CC(CC)C2CCC2)CC1.C1CCC1 C1(CNC(=NCC2(CO)CC23CCOCC3)NC2CC2)C(F)(F)C12CCOCC2 C1(NC(c2ccnc(C)c2)CCC)C2CN(Cc3ccccc3)CC12 C1(C(CC)(C)C)CCC(C(C(=O)NC)N(CCCC(=O)NC2CC2)C)CC1 C12(C(=O)NC(C(=O)NC3(CCOC)CCC3)Cc3ccco3)CCCC1C2(F)F C1(c2cc(C)no2)CN(C(=O)NCc2nnc(C(F)(F)F)s2)CCO1 C1(C(=O)NC2CCC(CNC(c3ccc(CN=[N+]=[N-])o3)=O)C2)CC2CCC(C1)O2 N1(C(C2(F)CCN(C(c3cc(SC)oc3)=O)C2)=O)CC(C#N)C2(CCC2)C1 c1(OC(CC)C(=O)NCCCCN(C)C(C2CC(F)C(=O)N2)=O)cccc(C)c1 c1(C(=O)OC)cccnc1NC1CC(NC(C2CCSC2)=O)C1 c1(CC)nc(C)c(C(N2CCCC(NC(=O)C(c3cccc(F)c3)C)C2)=O)s1 C1(NC(CNC(C(CC)CC)=O)=O)CCCN(C(c2onc(Br)c2C)=O)CC1 C1(C(=O)NCCCCN(C(C2(CCC)CCC2)=O)C)COc2ccc(F)cc2C1 C1(C)(C(=O)NC(C(C)O)CCO)CCN(C(=O)CCC2CCCCO2)CC1 c1(C(=O)NCC2CC(NC(C3C(C)(C)CO3)=O)C2)[nH]nc2c1CCCC2(C)C c1(C(=O)NC2C=CCN(C(CC(CCCC)O)=O)C2)nnc(O)c2ccccc12 CCC(C)CC(=O)NCC(C)(O)CNC(c1ccc(C(=O)NCC2CC2)cc1)=O C(=O)(C(=O)CCC(C)C)N1C(CC(=O)NCc2c(C)nn(C)c2)CC(C)(C)C1 c1(C(N(Cc2nc(C)sc2)Cc2ccccc2)=O)nccc2c(Br)cccc12 Cc1nnn(CC(N2CCC2CNC(=O)Cn2cc(C(C)O)nn2)=O)n1 c1(OC(C)C(=O)NCC2CCCN2C(=O)CC2CCC2)ccccc1F N1(C(C(CC=C)(C)C)=O)CCOC2CCN(C(=O)CSC(F)F)CC12 C1(CC)CN(C(c2ccn(C(F)F)n2)=O)CCN1C(c1ncn2c1CCC2)=O C(=O)(CCC(=O)N(CC(O)CC(=O)NC(CC)C(=O)NC)C)NCC C(C1CCN(C(C2CCCOC2C)=O)CC1)=CC(=O)NC(c1nn(C)cc1O)C c1(CC)ccc(NC(=O)NCC(N2CCOCC2)C)cc1CC.C(C)(=O)N Cc1sc(C(=O)NC2CCCC2NC(c2ccc(N)cc2F)=O)cc1[N+](=O)[O-] c1(SCCC(N2C(C)CC(n3ccnc3)C2)=O)ccc(F)cc1F N1(c2c(C)c(N(C)CCc3cccnc3)ncn2)CCC2OC(=O)NC2C1 C12(C(N(CCCCCNC(C(F)=CC)=O)C)=O)CCC(CO)(CC1)CC2 c1(C(N(CC)CC2(C(=O)OCc3cncc(Cl)c3)CC2)=O)cccc(S(N)(=O)=O)c1 C1(C2(O)CN(C(C3COCCN3C)=O)C2)(CNC(c2c(C)[nH]nc2CO)=O)CC1 C1(NC(=O)NCCCc2n(C)ccn2)CCN(CC2CCOC2)CC1 c1(C(=O)NC2CC3CN(C(C(C)C(F)(F)F)=O)C2C3)n[nH]c2c1CSCC2 N1(C(C(CC)(C)OC)=O)C(C)CC2CN(C(=O)CCSC(F)(F)F)CC12 c1(OCC)cccc(CN2CCC2(C)C(=O)NC2CCCC(CO)C2)c1Cl N#Cc1cc([N+](=O)[O-])cnc1NCC1CC(NC(=O)C=CC2CCC2)C1 CCCC(C(C(=O)NCc1ccccc1Br)N1CCCC12CCC2)OC C(=O)(C(C#N)CCN)N1CC(c2cn(-c3n(C)ncc3I)nn2)(N(C)C)C1 c1(NC(=O)NCc2nc[nH]n2)cccc(CN2CCNC2=O)c1 C1(CC(=O)NCC2N(C(COCCCC#C)=O)CC2)C=CS(=O)(=O)C1 C(CC(=O)N(C)CC1(CNC(=O)CCC2CCCCO2)CC1)(C(C)C)OCC c1(C(N(CCN(C)C(C2(O)CCCOC2)=O)C)=O)cnc(Cl)n1C c1(CC)c(C(N2CC(C(=O)NCc3[nH]nnc3C)C(CC)C2)=O)cnn1C C1(C(=O)NC2CC(CNC(C3C(C(N)=O)C3)=O)C2)CCn2nccc2C1 C1(C(=O)NCC2CCC(NC(c3n(CC)ccc3)=O)CC2)CCc2nn[nH]c2C1 c1(C(N2CC(NC(C=COCC)=O)C(F)C2)=O)c(Cl)cc(Cl)c2ncccc12 N1(C(C(C=C=C)C)=O)CC(NC(c2c(C)ncn2C)=O)CC2(CCC2)C1 c1(CC)ncc(C(N2CC(O)(C(C)NC(c3cnn(C4COC4)c3)=O)C2)=O)s1 N(S(=O)(=O)N1CCC(C(=O)N(C)C)CC1)(CC(C)C)C1CC1 Nc1c(C(N2CCOCC2CNC(c2cnsc2)=O)=O)cccc1F c1(CC)cnc(C(=O)N(CC(C)C(=O)NCCc2ccc(C(=O)O)[nH]2)CC)nc1 C1(NC(=O)COc2ccsc2Cl)CN(C(=O)CC2(CO)CC2)C2(CCC2)C1 C1(NC(c2c(C)con2)=O)C2CC(NC(c3c(C)ccn3C)=O)CC12 CCCCCC(c1nnnn1C1CC1CC)Nc1cnoc1 CCS(=O)CC(=O)NCC12CC(CNC(=O)C(C3CCCC3)OC)(CO1)C2 C(CN=c1nc2scnc2c(NC2CCC3(C2)CC3(F)F)[nH]1)SC N1(C(C(CC)(CNC(C2OCC3CCCC23)=O)CC)=O)CC2CCCCC2C1C c1(C(=O)NCC(CO)NC(=O)CCc2ccc(F)nc2)ccnc(N2CCC2)c1 C1(CC(C)C)(NC(=O)NC2(C)CC2C2CCCO2)CCCCC1 CC(CNC(c1ccn(C(F)F)n1)=O)C(=O)N1CC(n2cccn2)C1 N1(C(c2c(C#N)scc2)=O)CC2CC1CC2NC(c1cc2n(c1)CCC2)=O N1(C(C)=O)CCCC(C(N2CCC3C(NC(C4CCOCC4)=O)C23)=O)C1 C1(CNC(c2c(OC)n[nH]c2)=O)(NC(=O)C(C2CCCC2)OC)CCCCCC1 c1(C(N2C(C(C)NC(C3CCCC3(F)F)=O)CCC2)=O)cn2cccc(Cl)c2n1 C12(C(=O)NC3C(CNC(c4ccnnc4O)=O)CCC3)CCCC1C2(F)F c1(CCC)n[nH]c(=NC(C)CC(C)NC(c2cc(OC)ns2)=O)s1 C1(C(=O)NC2(CC=C)CN(C(=O)C(C)(C)F)C2)CCCCC1C1CC1 c1(CCNC(C(C2(O)CN(C(CC3(OCC)CC3)=O)C2)F)=O)ccc(C)nc1 C1(CNC(C(c2cnn(C)c2)OC)=O)CCN(C(=O)CC2(C#N)CCC2)C12CC2 C(C(O)C(C)(C)C)N(C)C(C1CCC(NC(C2(O)CCSC2)=O)C1)=O C(=O)(C(C)CC(F)(F)F)N1C(CC(=O)NC2CC(OCC)C2)CCC1 CCCCC(C(=O)N1CCCC(O)(CCNC(=O)C=C2CCSCC2)C1)N(C)C C=CCC(CNC(=O)C(F)C(C)(F)F)C(=O)NCCN1CCCOCC1 C1(C(N(CCCNC(c2n[nH]c(C)c2C)=O)C)=O)OCCN(C)C1=O C(N=c1[nH]c2ccc(Br)cc2o1)C1CC(C(CC=C(Cl)Cl)=O)C1 C1(NC(C=Cc2nnn(C)n2)=O)CC2CCC1N(C(=O)C1=CCCCC1)C2 N1(C(CC(=O)OC)=O)CCC2(CNC(c3cn4ccnc4cn3)=O)CCCCC12 Cc1ccc(C(=O)NCc2csc(C(=O)NC(CN(C)C)C(C)C)c2)cc1F C(=O)(CCCCCNC(N)=O)N1C(CCNC(C(CCC)C)=O)COCC1 C=C(Cl)CC(C(=O)NC(C(=O)N(C)C)C(C)C)NC(c1cn(C)nc1CC)=O N1(C(c2cc(CCC)n(C)n2)=O)CC2(CCCC2NC(=O)C(C)C(F)F)C1 N1(C(COCC(C)(C)C)=O)CCN(C(=O)C=Cc2ncco2)CC1CC(C)(C)C N1(CC)CCCC1CC(=O)NC1CC(NC(=O)C(F)(F)c2ccnn2C)C1 c1(OC)ccc(C)c(C(N2CCC(NC(=O)C3=CCS(=O)(=O)C3)C2)=O)c1N C1(NC(c2ccsc2Cl)=O)C2CC3CN(C(=O)C4CCc5c[nH]nc54)C1C3C2 C1(C(=O)NCC(CC=C)NC(c2cc(CC)on2)=O)CC2(CCC2)CCO1 c1(NS(C)(=O)=O)cccc(C(N2CCC(CNC(c3cc[nH]n3)=O)C2)=O)c1 C(=O)(N1OC2CCC1CC2)C1C(NC(C2(CC=C)CC=CC2)=O)CCOC1 C1(NC(Cc2c(C)occ2)=O)CN(C(=O)C(C)(C)C2CCC2)CCC12CCC2 CCC(C)CCNC(=O)C(CNC(=O)CC(C)=C(C)C)OC C1(CC(=O)N(CCC(=O)N(C)Cc2cnc[nH]2)CC#C)CCC2CC12 n1(CC(N2C(CNC(C3C=CCC3)=O)CC(OC)C2)=O)[nH]cc2c(=O)ncnc1-2 c1(CCC(=O)N(C2CCC(OC)C2)C)ccc(-c2cncnc2)cc1 CCC(C)(F)C(=O)N1CCC(CN(C)C(C2CCCO2)=O)CC1 c1(CC)cccc(C(N2CCCC(C(=O)N(CC)Cc3noc(C)n3)C2)=O)n1 N1(C(C2C(C#N)C2)=O)CCN(C(=O)CO)CC1 C(=O)(C(C)(C)CC(=O)NCC(C)(C)CNC(C1CC(C)(F)C1)=O)OCC O=C(CN=c1cc[nH]cc1)NC1CCC(CC(N2CCCC(O)C2)=O)C1 CC1(C)CCC(C(C)(C)C)N(C(=O)NC2CC2c2ccccc2Br)C1 C(C)(C)(CC(=O)N(C(C)C(F)F)C)C(C)C(=O)N.N(C)C C(=O)(C1CCCc2c[nH]nc21)NC(C)CCNC(=O)C=Cc1ccccc1F c1(C(C)NC(CCn2cc(-c3c(C(=O)OC)n[nH]c3)nn2)=O)nccc(O)n1 Cc1ccc2[nH]nc(C(=O)NCC34CCCC3N(C(C3CSC3)=O)CCC4)c2c1 N1(C(C(CN(C(=O)CC2CC=CCC2)C)(C)C)=O)CC2CC1CC2CF c1(OC)cc(Br)c(Cl)cc1NC(C1(C)CCN(Cc2cccc(C)c2C)C1)=O Cc1cc(CN2CCN(C)CC2C(N2CCOC(CO)C2)=O)c(C)cc1O C(CCC(O)C(=O)N1CCC(N2CCC2)CC1)NC(C1(C)CCC(=O)N1)=O O=C1NC(Cc2ccc(Cl)cc2Cl)C(=O)N1CCSC1CCCC1 CC(C)(C)C(C(=O)N=c1[nH]oc2cccc(F)c12)n1ccnc1 Cc1cc(C(=O)NCCC(O)CNC(=O)CCN2CCCC2=O)cc2ccoc12 C(=O)(C(F)(F)CC1CCCO1)N(C1CCN(C(=O)CSC2CC2)C1)C C(=O)(CCP(C)(C)=O)NCC1C(NC(CN(CC)CC)=O)C1(F)F Cc1c(C(N2CC3CC2(CNC(c2ccsc2)=O)C3)=O)sc2cncn12 N1(C(C(C)OCc2ccc(Cl)c(Cl)c2)=O)CCC2(C1)CN(C(=O)C(C)N(C)C)C2 C1(CC=C)(NC(=O)CNC(c2nn(C)c(C)c2Cl)=O)CCCN(C(=O)COC)C1 C(CC(=O)NC1(C(C)C)CC1)(C(C)CC)NC(CC(C(=C)C)OCC)=O c1(OC)ccc(F)c(C(=O)NCC2CC(O)CN2C(C2CCN(C)C2C)=O)c1F C(=O)(C1=CCC(C)CC1)NCC1C2CN(C(c3c(Cl)ncc(C)c3)=O)CC21 c1(C(N(CCN(C(C=C(C)C2CC2)=O)C)C(C)C)=O)cnn(CC2CCC2)c1 c1(C(=O)NCC(C(C)C)NC(C(CC)=CC)=O)cc2cc(OC)ccc2[nH]1 C1(NC(C2CC2F)=O)C2COCC1CN(C(c1cscc1I)=O)C2 C12COc3ccc(cc3C1)CO2.C1(C(N2CCOCC2)=O)CC(=O)C12CCCCC2 C1(CCNC(c2cncc(F)c2)=O)CCCN(C(C2CCCC2C(F)F)=O)C1 c1(C(=O)NCC2CN(C(C3N(C)CCOC3)=O)CC2(C)C)ccc2sccc2c1 C(=O)(C(C)CC)N(C1(C(=O)OC)CCC1)CC1CC1 C1(C(=O)NCCC(CC)(F)F)C(C)OCCN1C(C1CCCN1C)=O C(=O)(CC1=CCN(C)CC1)N1CCC(NC(c2c(OCC)nccc2)=O)C(CO)C1 N1(N2CC(C)N(C=O)CC2)CCc2c[nH]nc2C1.c1(C=O)ccn2ccccc12 C1(NC(=O)NC2C(OC)CC2)CCN(C(=O)CC(=O)Nc2nccs2)CC1(C)C C=C(C)c1ccccc1NC(=O)C(O)CCNC(c1nsnc1O)=O Cc1cc(C(=O)N(C2CN(C(C3CCOC3C3CC3)=O)CC2(C)C)C)cc(Cl)c1 N(C1CCCn2ncnc21)C(C1C(CNC(C2(Cl)C(C(C)=O)C2)=O)C1)=O c1(N2CCN(C=O)CC2)snc(C)c1C#N.c1(N(CCC)CCC)cnn(C)c1 C(=O)(CC(C)(C)C)NC(C1CCN(C(=O)NC2CCCN2CC(F)(F)F)C1)C Cc1cc(=O)oc(C)c1C(=O)NC(C)CCNC(C1CCCC2C1C2(F)F)=O c1(C(=O)NC2CC3CC(NC(=O)CC45CCCC4C5)C3C2)ccn2nnnc2c1 N1(C(=O)NC2C(C)CCC2)CC2CCC1CN2C(c1csc(CO)n1)=O CC(=O)CCCC(=O)N1CCN(C(=O)Cc2ccnc(F)c2F)C2CC12 C1(NC(c2c[nH]nc2C2CCC2)=O)CC2CCC1N(C(=O)CN1CCSCC1)C2 N1(C(c2cccc(Oc3cnc[nH]3)c2)=O)CCCCCC1CCO N1(C(c2ncc(CSC)o2)C(=O)Nc2ccc(Cl)cc2F)CCCC(F)(F)CC1 c1(C(N2C(Cn3cc(C(COC)O)nn3)C(C)(C)C2)=O)ccnc2c1ncn2C N1(C(C(C)=CCC)=O)CCCC1C=CC(=O)NCc1coc(C)n1 N1(C(c2ccc(OC)cn2)=O)CCN(C(C2CC23CC3(F)F)=O)C2(CCC2)C1 C1(NC(CSCCC)=O)CCN(C(=O)C(C)C2CC2)C1C(C)C c1(C(=O)NCC2N(C(COCC(C)C)=O)CCC2)ccnc(OC(F)F)c1 c1(CCC)cc(=NC(=O)N2CCCC2C)[nH]o1 C1(NC(=O)CSCc2ccccn2)CCN(C(c2cc[n+]([O-])cc2)=O)CC1F c1(CCC)[nH]nc2ccc(C(=O)NC3CC(C)(CNC(C4CC4C)=O)C3)cc12 C(=O)(C(CC(F)F)NC(c1cc(CO)n(C)n1)=O)NC(CC)CO c1(C(N(c2nccc(Br)n2)C2CC(N)C2)=O)cnc2ccccc2n1 C12(COC)CC(CNC(c3ccccc3)=O)(CN1C(C1CCC(C#N)CC1)=O)C2 c1(OC)cc(C(=O)NC2CCC(CCNC(=O)CN(C)C)C2)cc(C)n1 C1(NC(C(COC)C)=O)CN(C(c2nnc(O)cc2O)=O)CC12CC2 C(C)(C)(CC(F)C(=O)N1CCC(CO)=C(F)C1)NC(CC(COC)C)=O C=CC(C)C(C(=O)OCc1ccc(F)c(F)c1)c1ccccc1 C1(C(N2CC3C(CNC(CC4CC(=C)C4)=O)(C3)C2)=O)CCN(OC)CC1 N1(C(CCc2ccc(C)s2)=O)CC(NC(=O)CC2(N(C)C)COC2)CC1(C)C c1(CC(=O)NCC=CCC(=O)NCC2CC(CC)C2)c(C)noc1C c1(C(=O)NCC(CNC(C2C(C)C2C)=O)C)ccoc1C1CC1 c1(N2C(C(=O)Nc3cnn(CC(F)F)c3)CC(OC)C2)ncnc2n[nH]c(Br)c12 N1(CCCC)CC(C(=O)NC2CC(NC(=O)Cc3nc[nH]n3)C(O)C2)CC1=O c1(C(=O)NC2CC(CNC(CC3(O)CC(C)(C)OC3)=O)C2)ccc2[nH]ccc2c1 Cc1[nH]c(=N)ccc1C=CC(=O)N(CCNC(=O)COc1ccn(C)n1)C(C)C c1(C(N2CC3C(NC(C(CC(C)C)C)=O)(C3)C2)=O)cnn2c1OCCCC2 c1(C(N2CCC(NC(c3coc(C4CC4)n3)=O)C2)C)cccc(Cl)c1 C1(C(N2CCC(N(C)C(c3cnn(CC(F)F)n3)=O)CC2)=O)CCC(C#N)CC1 N1(Cc2c(C)occ2)C(=O)CCN(CC2CCCCN(C)C2)C1=O CS(=O)(=O)C1CCCC1C(N1CCC1CNC(=O)CC1CC(C2CC2)C1)=O c1(CC(=O)OC(c2ccc(OC3CCN3)nc2)=O)ccc(OCC(F)(F)F)nc1 C1(CC)CCC(C)CN1C(=O)CCN(C(=O)CCC1CC1(F)F)CCO N1(C(C(CC#C)C)=O)CCCC2(CCCN2C(c2ccnc3ccnn23)=O)C1 c12ccc(cc1Cl)COC(=O)C1CC(C)CN1C2=O.COC C(=O)(C(C)CC(=O)OC)NCC1CCCN(C(Cc2ccc(OCC)cc2)=O)C1 c1(C2(C(=O)NC(C(C)C)CNC(=O)C=CC=CCO)CC2)cccc(F)c1F c1(C(N2CC(C)C(NC(C3CC4C=CC3CC4)=O)C2)=O)nccc2c1CNC2=O C1(C(=O)OC(C)(C)C)CN(C(c2ccc(-c3cnco3)cc2)=O)CC1(C)C C1(c2nnnn2C2COC2)(Nc2c(C)ccc(C(N)=O)c2)CC2CCC1CC2 Cn1c(O)nc2cccc(C(=O)NC3CC(NC(=O)C(C)(C)C(F)(F)F)C3)c12 n1(CCCCNC(CC2(CSC)CC2)=O)cc(Cc2nc(C)no2)nn1 Cc1nc2sccn2c1C(=O)NCCC1(NC(C2CC3(C2)CC(O)C3)=O)CCC1 C=CC(C)(O)C(=O)N1CCC(C(C)(C)CNC(C2C3CCCC23)=O)CC1 Cc1cnc(C(C)NC(=O)CC(C2CC2)NC(=O)C(C)OC(C)=O)nc1 C(=O)(C#CC1CCCOC1)NCCCN(C(=O)CC1CCCC1)CC c1(OCC)cc(C(=O)N(c2cc(F)cc(F)c2)CC)cc(Br)c1OC c1(C(=O)NC2CCC(C(=O)NCC3CCO3)C2)ccc(C(F)(F)F)c(Br)c1 Cc1cnc(C=CC(N2CCCC2CCNC(=O)CC2CCC(F)(F)C2)=O)[nH]1 c1(N2CC(CC=C)(NC(=O)C(C)C3CCC3)C2)nc2ccc(C)nc2s1 CC1CC(NC(=O)C(CO)N(C)C)CCN1C(c1ccnn1C)=O OC1CCCCC1CNC(c1nnnn1CCC1CC1)c1ccno1 C1(C(=O)NC(c2cccnc2)C)CCCCC1NC(=O)C(O)c1ccsc1 C1(CNC(c2cc(C(=O)OC)nn2C)=O)(OC)CCCS1(=O)=O c1(C(C2CCCN(C)C2)C(=O)NCCC(C)OC)cnc(N2CCCC2)nc1 c1(C(=O)NCC23N(C(Cc4cn(CC)nn4)=O)CC(C2)C3)ccc(F)cc1Cl c1(C(=O)NC2(C)CCCN(C(c3cc(C)oc3C)=O)C2)ccc2c(c1)C=CCC2 C(=O)(C(C)(F)C(C)(C)F)N(CCN(C(=O)Cn1cc(C(F)(F)F)nn1)CC)CC CC1CCCc2nc(C(N3CCC(C)(CNC(C4(CO)CC4)=O)C3)=O)cn21 c1(NC(C(=O)NCC(C)N(CCC(C)OC)C)=O)c(OC)ccc2ccccc12 N1(C(CCC)=O)CC2CCC1C(NC(c1ccc(C(N)=O)o1)=O)C2 C1(C(=O)NC(C2CCOC2)C#C)CCCCN(C(c2c[nH]cc2CC)=O)C1 C1(CC)CC1(C)C(=O)CCNC(=O)CN(C)C(C1CC1C(=O)OCC)=O c1(C(C)=O)ccc(C(=O)NC2CCCC2NC(=O)C(C)(COC)OC)cc1F Cn1cc2ccc(C(N3CCN(C(=O)C=Cc4ccc[nH]4)C(CO)C3)=O)cc2n1 c1(CC(=O)NCC(C(C)C)(C)NC(c2ccc(O)nc2)=O)cccc(Cl)c1F C1(C(N(C2CC2)CC2N(C(C3CN(C(C)=O)C3)=O)CCC2)=O)CCCC2(CC2)C1 N1(C(c2occ(C)c2)=O)CCSCC1C(=O)NCC1(CC2CC2)CCC1 Cc1cc(NC2CC(NC(c3cc(O)nn3C)=O)C23CCC3)ccc1[N+](=O)[O-] c1(C(N2Cc3c(nc(C)[nH]3)CC2)=O)ncnc2ccc(N3CCOCC3)cc12 CC1C(C)N(C(=O)CCOCC2CCCC2)CCN1C(=O)CCCF C1(C(=O)NCCCOC(C)C)CN(C)CCN1C(=O)Cn1cccn1 c1(COC)ccnc(F)c1-c1nc(C(=O)Nc2ccc(O)cc2F)cs1 C1(O)(C(=O)NC2CC(NC(C(C)Cn3cccn3)=O)C2)CCCCCC1 CCC(C)(C(=O)O)N(C)C(c1ccc(-n2cncn2)cc1)=O C1(NC(COC)Cc2ccccc2)CCCN(Cc2ccccc2)C1 c1(C(N(C)CC2CCCN(C(C3CC3C(C)(F)F)=O)C2)=O)cc2c[nH]cnc-2n1 C1(C(C)NC(C(CC)N(C)C)=O)CN(C(C2CN(CC)CCO2)=O)CCO1 c1(C(N2CCC(CCNC(=O)C(F)OC(F)(F)F)C2)=O)cc2ccccc2cn1 C1(NC(CCOC)=O)CC12CCN(C(C1CC(=O)N(C3CCCC3)C1)=O)CC2 CC1(C(=O)NCC2CC(F)(CNC(c3csc(CO)n3)=O)C2)CC(F)(F)C1 c1(CCNC(c2n(CCCC)nnn2)(C2CCCCO2)C)cc(Br)ccc1F c1(CNC(c2cc(-c3cn[nH]c3)ccc2CO)=O)ccc(Br)c2ccccc12 C(C)(C(=O)N(C(C)C(=O)N(C(COC)C(C)C)C)CC)O.CC(=O)NC c1(C(=O)Nc2nc(C(=O)Nc3cc(Cl)ccc3Cl)cs2)cccc([N+](=O)[O-])c1 C(=O)(CCCC(=O)N1CCCC(NC(c2[nH]cnc2C)=O)C1C)OCC Cc1cc(C(C)NC(c2cn(CCNC(=O)Cn3ccnc3)nn2)=O)no1 C(=O)(C(CCF)NC(=O)Cc1ccc[nH]1)NCc1[nH]nc(OC(C)(C)C)n1 C1(O)(C(C(=O)NC(C)C(C)N(C)C)NC(Cc2nc(C)sc2)=O)CCCCC1 N1(CC)CCOCC1C(=O)NC1CCC(F)(CNC(=O)CCc2scnc2C)C1 C1(OC)C(OC)CN(C(=O)CN(C)S(N)(=O)=O)C1CNC(C1CCCCO1)=O C(C(O)CCCS(N)(=O)=O)NC(CS(N1CCN(C)CC1)(=O)=O)=O Cc1ncnc(NCc2cn(CC3CCCN3C(C)=O)nn2)c1C.C(C)(C)(C)NC=O C(C)(C(=O)NNc1cccc2c1OC(F)(F)O2)(C(C)C)OC C(=O)(CC(O)(C(F)(F)F)c1ncc[nH]1)NC(C)C(C)(C)NC(c1cnnc(O)c1)=O C1(NC(C2C(C)OC(C)C2C)=O)CC2(CCCCN2C(C2CCC3CC3C2)=O)C1 c1(Nc2ccccn2)nc(N(CCCCC=C)C)c2c(F)cccc2n1 C1(C2CN(C(=O)COCP(C)(C)=O)C2)(NC(C2CC(C)CC(C)O2)=O)CC1 c1(C(N2CC3C(CN(C(=O)CCC4CC4)C)C3C2)=O)ccsc1S(C)(=O)=O c1(OCC(=O)NC23CC(CNC(C4CCCOC4)=O)(C2)C3)ccc(F)cc1F NS(=O)(=O)CCNC(=O)CCNC(C1CC(NC(=O)C(F)C2CCC2)C1)=O c1(C2C(=O)N3CCCC(C3)N2C)ccc(Cl)cc1.S(=O)(=O)(C1CC1)N.CN N1(C(C2CCCC2)C)CC2CC(C(=O)NCCC3CC3)CC1C2 C#CCC(C)(CNC(c1cc(CNC(=O)CC(C=C)CC)nn1C)=O)CO CC1CN(C(c2sccc2F)=O)CCC1NC(=O)Cc1cncn1C CCCCC(C)C(=O)NC1CN(C(c2ccnn2CCC)=O)CC1CC1CC1 C12(C(=O)NCCOCCNC(c3cn(CCC)nn3)=O)CCC(OC)(CC1)C2 Cc1nn(CC(N2CCC(C)(NC(C3CC3C#N)=O)C2)=O)c(C)c1Cl n1(CC(=O)NC23CN(C(c4ccc(N)cc4F)=O)C(C2)C3)ncc2ncccc12 c1(C(N2CCCC(NC(c3c(C)nc(C)s3)=O)C2C)=O)cccn2c(C)cnc12 C1(NC(Cn2ccc(C)n2)=O)CC2(C1)CC2C(=O)N(C)CCc1nc(C)cs1 C=CCC(C)(O)C(=O)N1CCCC(NC(=O)COCC)CC1 C1(NC(C2CC(C)(C)C2)=O)CC(Nc2ccc(CCn3ccnc3)cn2)CC1O N1(C(c2ccn(C(C)(C)C)n2)=O)CC(NC(=O)C(N)=O)CC12CCC2 c1(NC(=O)C2CC2)cc(Nc2cc(OC)cc(NCSCC)c2)ccc1C N1(CC)CC(C(N2CCC(OCCNC(=O)C=CC(N)=O)C2)=O)CCC1=O N1(C(C(C2CC2)OC)=O)CCC2CC(C1)CN(C(C1CN3CCN1C(C)C3)=O)C2 CN=c1nc(N2CCCC(C)(F)C2)[nH]c(=NCC2=COCCO2)[nH]1 CC(C)C1=CCC(C(N2CCCC(N(C)C(C3CC(F)(F)C3)=O)CC2)=O)CC1 CCC(CNC(=O)C(F)CC1CCC1)C(C)C.C(=O)(CCC)N1C(=O)C1 c1(OC)cccc(NC(=O)NC(Cn2ccnn2)C(=O)NCC(O)C(F)(F)F)c1 CC(C)C(C)(O)C(=O)N(CC(C)NC(C1CC1C(N)=O)=O)C c1(OCCC)ccc(Cl)cc1C(=O)NCC1(C)CCC(NC(c2cn[nH]c2)=O)C1 C1(C(=O)NCCN(C)C2CC2)CN(C(=O)Cn2ncnn2)CCO1 C(C)(CCC(=O)C(=O)CCC(C)N(C)C)SC.C1(N)C2CC(NC=O)CC12 N1(C(C(C)CO)=O)CCC(CC(C)NC(c2ccoc2Cl)=O)CC1 C(=O)(C(CO)N(C)C)N(C1CCCC1)CCCOCCNC(C=C(C)C(C)C)=O Cn1cc(S(N)(=O)=O)cc1C(N1CC(NC(c2ccc(N)cc2O)=O)CC1F)=O C1(C2CC2)(NC(CCC(=C)Cl)=O)CCN(C(c2cnc(OC(C)C)cn2)=O)C1 N1(C(C)Cc2ccc(C(F)(F)F)cc2C(F)(F)F)CCNC(C)C1C CN1CC2(CN(CC3CCOC3(C)C)C2)OCC1=O C(=O)(C(F)(CC)C(=O)OC)NC(CN(C(c1cc(CC)sc1)=O)C)C C(CC(C(=O)N1CCCC(CF)C1)NC(c1nc(=N)cc[nH]1)=O)OCC C(CCCCC(=O)N1CCC(C)(CCNC(c2[nH]cnc2C)=O)C1)=CCCC CCC(C)C(C(=O)NC)NC(=O)CCCNC(=O)CC(C)COC N1(CCC(=O)NCC)CCCC(C(=O)N(C)CCc2ccc(Cl)cc2)CC1 C1(C2CC2)(NC(=O)NCCC(COC)(C)C)CCCC1 CC1(C)CCC(=CC(=O)NCC2CN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)CC1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(C)Br)cccc2ccn(C)c12 C1(C(C)C)CN(C(c2ccc(C#N)cc2)=O)CCCN1C(=O)COC1CCC1 c1(NC(C2CCN(C(C(C)OC)=O)CC2)C)cccc(C)c1C C1(CC(=O)NCCCC2(NC(c3ccc(O)cn3)=O)CC2)CCCC2(CCC2)O1 Cc1cc(=O)ccn1CC(=O)NC1C2CN(C(=O)CSc3ccccc3Cl)CC12 c1(C(N2CCC(C(C)NC(CC=CC)=O)C2)=O)ccc(Cl)c(C)c1 N1(C(c2c(CC)noc2)C(=O)NCC2(CC)CC2)CCn2ncc(SC)c2C1 c1(COCC(=O)N(C(C2CCCO2)C)C)cn(C2COCC2O)nn1 C1(C)(C(=O)NCCCN(C(c2c(C)noc2C(F)(F)F)=O)C)CCCS1(=O)=O c1(C(=O)NC2(C(C(=O)NCCCC(=O)N(C)C)F)CC2)ccccc1F C1(CC(=O)NOC2CC2)C2CCC(C2)N1C(=O)Cn1nccn1 C1(NC(=O)COCC(F)(F)F)(CO)CCCN(C(C2CC3(CSC3)C2)=O)C1 C1(CC(=O)NC(CN(C(C2CC(C)SCC2)=O)C)C)CS(=O)(=O)CCN1C C(=O)(C(F)(F)CCn1cccn1)NC1CCC(NC(C2(C)C=CCC2)=O)CC1 Cn1cc(N)c(C(=O)NC2CN(C(=O)COc3cccc(C(N)=O)c3)CC2F)n1 Cc1cc(=O)cc(C)n1CCCC(N1CCCC(NC(=O)CCC(C)C)CC1)=O N1(C(CCCOC)=O)CCC(CO)C(NC(=O)Cc2cnccc2Cl)C1 c1(SC)nc(=NCC2(NC(c3cc(COC)[nH]n3)=O)CCOCC2)s[nH]1 c1(C(N2C(C)CCC(NC(=O)Cn3cnnc3O)C2)=O)sc2ccccc2c1Br Cn1nc(C(N2CC3CCN(C(=O)C(F)F)CCC3C2)=O)c2cc(F)ccc12 c1(C(N2C(CCNC(c3c(C)cco3)=O)COCC2)=O)[nH]c(=N)ccc1C C1(C(=O)NCC(CN(C)C(c2cscc2F)=O)(C)C)CCC2(CC1)CC2(F)F C1(NC(CC(C)OC)=O)CC(OC)CN(C(c2nn(C)cc2C)=O)C1 C(=O)(CCCC(C)(C)NC(C1CCC(C2CC2)C1)=O)NC1CC(C#C)C1 C1(NC(c2c(NC(C)=O)cncc2)=O)CN(C(=O)CCC(N)=O)C2(CCOC2)C1 c1(C(N(CC(C)NC(=O)C(O)CC2CCCC2)C)=O)coc(C(C)(C)C)n1 N1(C(C(CC)C(C)O)=O)CCN(C(c2cccc(C(F)(F)F)c2N)=O)C2(CC2)C1 c1(C(N2CC(CNC(c3ccccc3Br)=O)OCC2)=O)cc(Cl)ccc1Br N1(C(CC(CNC(C(CCC=C)(C)C)=O)OC)=O)C2CCCC1CC(=C)C2 Cc1ncccc1CN1CCN(C(c2cc(C3CCOCC3)on2)=O)CC1 C1(NC(C2(C(F)(F)F)CC(=C)C2)=O)CCN(C(c2ncc(F)cn2)=O)C1C1CC1 c1(C(=O)NCC2CCN(C(c3cnc(C(C)=O)s3)=O)C2)cccc2c1SCCC2 C1(C(=O)NCC(C)(C)n2ccnc2)CN(C(c2cc[nH]c2)=O)CC1C1CC1 c1(C(N(C2CC(c3ccc(C)cc3)C2)C=O)=O)nnn2c1CSCC2 N#Cc1cccc(NC(=O)CCC(N)=O)c1.C(c1cscn1)=CC(=O)N1CC1 c1(CN2CC(CC(=O)OCC)C3(CC2)CCC3)c(C)c2ccc(N)cc2oc1=O N1(C(C2CN(C)C(=O)C2)=O)CCCC(F)(NC)CC1.C12(C(=O)NC)CSCC1C2 C1(C)(CNC(C2CC(C)C2)=O)CCCN(C(=O)CCOC2CC2)C1 S(=O)(=O)(c1cnc(COC)s1)NC1(C)CCC1.N1(CCN)CCOCC1 Cc1c(CCNC(=O)C=CC2CCCN2C(C2CC(CF)C2)=O)cnn1C C1(C(N(CCNC(CC(=O)NCC)=O)C2CC2)=O)CCOC(=O)CC1 c1(CC)nnc(S)n1CC(N1CCCC(CN(c2ncnc(=N)[nH]2)C)C1)=O S(=O)(=O)(c1ccc(Cl)c(C(=O)NCCCC2(C)CC2(F)F)c1)N(C)C CC1CC(NC(=O)C#CC2CC2)CN(C(c2nc(C3CC3)ncc2Br)=O)C1 S(=O)(=O)(c1ccc(Cl)cc1F)N(C(C(CCC)C)C)CCO c1(C(=O)NC2C3(CCN(C(CSCC)=O)C3)C2)ccccc1S(=O)(=O)N(C)C C(=O)(CCCCCNC(=O)CC1CCOCC1)N1C(CC(N)=O)CCC1 C=CC(CCC)CC(=O)NCC12CC1CN(C(=O)COc1cccc(F)c1)C2 C1(NC(C(c2cccc(C)c2)(F)F)=O)CC2CCCC(C1)N2C(C1CC1C)=O c1(C(=O)NC(C(C2CC2)OC)C)cc(Br)cc(S(C)(=O)=O)c1F c1(C(=O)NC(C)CN(C)C)n[nH]c2c1CCN(Cc1cc(F)c(F)cc1O)C2 C(C(C(C)C)C1CC1)(OC)NC1CCCC(CO)C1 c1(C(N(CCNC(c2nccn2C)=O)CC)=O)cc(C(=O)OC)ccc1C c1(-c2cn(CCN(C(=O)COCC3CCCO3)C)nn2)cccc(N)n1 N1(C(c2cc(CC)nn2C)=O)CCC12CN(C(C1(C)CCCC1)=O)C2 c1(C(N(C)CC2(CNC(c3cscc3C(F)F)=O)CC2)=O)nnc(O)cc1O CN1CC(C)(C(=O)NCC2(F)CCN(C(C3CC3C(F)F)=O)CC2)CCC1=O c1(SC)ccc(C(=O)NCCc2cn(CCc3cccc(F)c3)nn2)c(Cl)c1 C#Cc1cccc(C(=O)NC(c2ccccc2)CNC(c2cocc2C)=O)c1Cl c1(C(=O)NC(C)CCNC(c2ccc(C(C)(F)F)nc2O)=O)cccc(F)c1N N1(CC#CCC)CCCC(COC(=O)CC2CCCCC2)C1 CC1OC2(C(=O)NCC3(CNC(C4CSCCS4)=O)CC3)CCC1CC2 Cc1nc(CNC(=O)C(C)NC(=O)Cc2coc(C)c2)co1 c1(NC(C2N(Cc3c(C)cc(Cl)c(Cl)c3)CC2)=O)c(C#N)ccc(F)c1F c1(CC(=O)NCC(C)(C(C)C)NC(C(C)NC(CC)=O)=O)cccc(C)c1Br C(CC(C(=O)N(C1CCCC1)C)NC(=O)C(O)Cn1cncn1)=CC c1(OCC)ncc(Br)cc1C(=O)NCC(CNC(=O)CSC)OC(C)=O C1(NC(C(C)CC2CCC2)=O)CCN(C(=O)C2CC2)C12CC2 c1(NC(c2cc(C(=O)OCC)n[nH]2)=O)ccc2c(c1)n(C)c(=O)n2C C(=O)(C(C)C(O)C(C)C)N1CC2C(CN(C(c3c(OC)cncc3)=O)C)C2C1 N1(C(C2C(C)(C)CN(C(=O)COCCF)C2)=O)CCOC2COCC2C1 c1(N2C3CC(CNC(C4C(CC)OCC4)=O)(OC3)C2)nc(C)nc(C)c1F c1(CC)cncc(C(N2CC(CNC(c3ocnc3CC)=O)C(C)C2)=O)c1 CC(C)CC(F)(F)C(=O)NCC(C(=O)NCCF)NC(=O)CN1CCCOCC1 C1(CNC(C=CC=CCC)=O)CC(C(=O)NC(C)C(=O)N(C)C)=NO1 N1(C(CCCCOCCC=C)=O)CC(CNC(c2ccc(SC)o2)=O)C2(CC2)C1 C1(CC(C)NC(=O)Cn2cc(-c3ccccn3)nn2)CCN(C(=O)CNC=O)CC1 C#Cc1ccc(C(N2CC(OC)C(C(=O)NC3CC(CC(N)=O)C3)C2)=O)cn1 C1(OC)CN(C(c2cnn(CCO)c2)=O)CC1NC(=O)CCN1CCCCC1C C(C(=O)NCC(O)CCNC(C1CCCOC1)=O)(C(C)C)SCC C1(NC(C2CCN(C(C)=O)C2)=O)CC2(CCN(C(c3cccc(=O)n3O)=O)CC2)C1 c1(CC)ccc(C)c(C(N2CCCC2C(C)NC(C2CCCN2CC)=O)=O)c1 N1(C(c2c(COC)cccc2)=O)CCC(NC(C2(CCN(C)C)CC2)=O)C(C)C1 C(=O)(CC(C)(C)C(F)F)N(CCNC(C1COCC(C)O1)=O)CCOCCO N1(C(Cn2c(C)csc2=O)=O)CCN(C(=O)COc2ccsn2)C(C)C1 C1(CNC(C(COC)(C)C)=O)CCN(C(c2n[nH]cc2C(C)(C)C)=O)CC1C c1(C(N(CCOC)CCNC(C2CNC(=O)C2)=O)=O)cc(F)cc([N+](=O)[O-])c1N Cc1ccc2nc(C(=O)Nc3cncc(-c4ccc(F)cc4)c3)ccc2c1 CC1CN(C(=O)C=C(Cl)Cl)CCC1NC(=O)CCc1cncnc1O c1(C(=O)NCCCOCCN(C)C(C2CC2C(C)(C)C)=O)ccc2ncnn2c1 C(CN=C(NCCN1CCCC1)NC1CCOC(C)C1)c1c(C)noc1C CC(C)CCCC(C)C(=O)NCC1(C)CCC(NC(=O)CCc2nc[nH]n2)C1 C(=O)(CCCN=c1nccc[nH]1)NC(CNC(C(C)NC(=O)NC)=O)C c1(NC(CCc2c(C)noc2)=O)cc2c[nH]nc2cc1F.C12CCN(CC1)C2=O C1(C)(CNC(CCOCCOCC)=O)CCCN(C(=O)CCC2CCC2)C1 N1(C(Cc2cc(C)c(F)cc2)=O)CCC(NC(=O)CCOCC(C)C)C12CCC2 C1(C(=O)NCCC(C)N(C(=O)Cc2ccnc(O)c2)C)CCC(O)CN1C CC(C)CC(C(=O)NCC1CC(C2CC2)CO1)ONC(c1cccn(C)c1=O)=O C1(CC)CN(C(c2cncn2C(C)C)=O)CCN1C(c1cccnc1S)=O c1(C(=O)NCCC2CCN(C(C3CCCN3C3CC3)=O)C2)cc2cccn2cn1 C(CC(C)C(=O)NCCOC1CN(C(C2CC23CC(O)C3)=O)C1)=CCC C(C(=O)NCC(C(=O)C1CC1)C1C(COC)C1)(C(C)C)OC.C12(CC1)NC2 c1(-c2scc(C(N(CCNC(C3(C)CC3C)=O)CC)=O)n2)ccccc1Cl C#CCCCC(C)C(=O)N1CCN(C)CC1C(=O)N(C)Cc1ccc(O)cc1 c1(C(N(C2CCCCC2)CCNC(C(C)N(C)C)=O)=O)nn[nH]c1Cl C1(NC(C(Cn2ccc(C)n2)C)=O)CC12CCN(C(C1(C)C=CCCC1)=O)CC2 O=C1COC(CNC(c2cn(CNC(C3(O)CC3)=O)nn2)=O)CN1 C(CC(C)CN=C(NCC1CC1)NC1CCN(S(C)(=O)=O)C1)SC Cn1cnc(C(=O)NCCCNC(C2CC(O)(CCC(C)(C)C)C2)=O)c1 C1(C(C)C(=O)N(CCCNC(=O)Cn2cccn2)C)CCOCC1 C#Cc1ccc(C(=O)NCC2CN(C(c3oc(CC)nc3C)=O)CCO2)c(C)c1 N1(C(c2ccnc(OC)n2)=O)CCC(c2ccccc2)(C(=O)OC(C)(C)C)CC1 C1(C(CNC(C2C(C)C2C)=O)(C)C)CCN(C(C2CCCC2)=O)CC1 C(C(C)C)(C(O)C(=O)NC1(CN(C)C(C2CC(F)C(=O)N2)=O)CC1)OC CCC(CC(F)(F)F)NC(=O)NC(c1ccc(F)cc1)c1cn(C)cn1 CC1C(NC(c2nonc2N)=O)CCCN1C(C1CC12CCOC2)=O c1(OC)cc(C(=O)NC(C)(C)CCN(C)C(C2OCCN(C)C2=O)=O)cnc1O C=CC(CC)C(=O)N1CCCC(CCC(=O)N(C)Cc2cnco2)C1 c1(NC(C(COC)NC(=O)C(N2CCOCC2)C)=O)cncc([N+](=O)[O-])c1 C(C)(CC(C)C)(C(=O)NC(C)CO)NC(CC=C=C)=O CCCN=C(NCC1(C)CCN(C)CC1)NC1CC(C(=O)OC)c2ccccc21 CC(O)C(C(=O)N1CC(CO)(NC(=O)C=CC2CCC2)C1)NC(=O)C1CC1 C1(OC)CCCN(C(c2cccc(-c3ccccc3)c2)C(=O)NC(C)C)CC1 C1(CC)CN(C(C2CCC3CC23)=O)CCN1C(=O)CCc1ncccc1C c1(CN2CC(N(C(C3N(C(=O)OCC)CCCC3)=O)C)C2)cnc2ccnn2c1 C(C)(CCC(=O)NCC(C)NC(=O)C(C1CCCCCC1)F)OC c1(C(=O)NCCCC2N(C(COCC(=O)NC)=O)CCC2)nc2c(s1)CCCC2 Cc1cc(NC(=O)COC2CCN(C(C3CCCN3C)=O)C2)cc(F)c1 Cc1cnc(CC(=O)N(C)C(c2cccnc2)=O)s1.C1C(O)CNCC(=O)N1 C(=O)(C1OCCn2ccnc21)N1CC(C)CN(C(=O)C=Cc2cccn2C)CC1 C=C(C)C(C)(C)C(=O)NCC1CCN1C(=O)C=Cc1cncc(F)c1 c1(C(CSCC)C)cn(CC2CCN(C(=O)CCc3ccccc3)C2)nn1 c1(C(=O)N)cc(N)cc(SC)n1.C1(C2CC2)C(=O)N1.C12CC1CNC2=O.CCOCC N1(C(c2c(SC)ccc(N)c2)=O)CCC(C2CC2)(NC(C2CCCN2CC)=O)C1 C1(NC(c2c(C(C)C)nco2)=O)CCC(O)CN(C(=O)C(F)C(C)(C)O)C1 C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)C(F)=C(C)C)CCC1CO n1(CC)ncc(C(=O)NCCC2(O)CCN(C(c3ccnc(SC)c3)=O)C2)c1Cl C(C1=NOC2(CCC2)C1)SCc1cn(C2CC(C(N3CC(C)OC(C)C3)=O)C2)nn1 CC1(C(N2CC3CC3(C(=O)NC3CCCC(C(N)=O)C3)C2)=O)CCNC1=O c1(C(=O)NC(C2N(C(C(C(=O)OC)C)=O)CCC2)C)cc2n(n1)CCNS2(=O)=O C=CCC(C(=O)N1CCCCC1CC=C)NC(=O)COCCSC N1(C(c2scc(C)c2)=O)CCC(C2(NC(=O)C(O)C3CCC3)CC2)C1 C1(Cl)(C(=O)NCC2(F)CN(C(Cc3nc(C)sc3)=O)C2)CC12CCC2 C1(C(C(=O)OC)N2CCC2)CC12CCC2 c1(CC)c(OC)cccc1C(=O)NC1CN(C(C2CN(C(C)=O)C2)=O)CC1(C)C N#Cc1sccc1C(N1CCC(CCNC(=O)C(C2CCOCC2)F)CC1)=O O=C(C1CCCn2ccnc21)NC1CC1CNC(c1cccc(Br)c1Cl)=O C1(NC(C2(C)CC2(Cl)Cl)=O)CC2(C1)CC(NC(C1COCCC1(F)F)=O)C2 Nc1c(C(=O)NC2COCC2NC(C2(CC(F)F)CCNC2=O)=O)ccnc1Cl N1(C(=O)CC2CC3(CC3)C2)CCN(C(C2C3CC4C(C3)C24)=O)C2(CCC2)C1 c1(C(N(C2CCCN(C(CNC(C)=O)=O)C2)C)=O)ccc(Br)c(Cl)c1 C1(C(=O)NCCOCCN(C(c2ncc3c(n2)CCC3)C)C)CCC2CCCCN12 S(=O)(=O)(C1(c2cn(CC3(Sc4cccc(I)c4)CCC3)nn2)CC1)N(C)C c1(N2C(C(=O)NC(CC)CO)CCC2)ncccc1Cl C(CCC(O)C(=O)N1CCC(CC2CCC2)C1)NC(CCC(C)OCC)=O CCC(CC(=O)NC(C)CCCNC(c1cc(C)n(CC)n1)=O)C(F)F N1(C(C(NOC)=O)=O)CC(C)OC2(CCN(C(=O)C(C)CS(C)(=O)=O)C2)C1 C1(CC(CC)NC(=O)C(CNC(=O)OC(C)(C)C)CO)CCCN(C)C1=O.C(C)(=O)O C#CCC(C(=O)NCCC(O)CO)NC(=O)C(C)C=C N1(C(C2CCN(C(N(C)C)=O)CC2)=O)CCN(C(c2csc(Cl)n2)=O)CC(O)C1 C(=O)(C(C)(C)CC(=O)OC)NC1CC(F)(CNC(C2(CCCC)CC2)=O)C1 n1(CC(N2Cc3ccccc3C2)=O)ccc(=NCc2c(Cl)cc(Cl)cc2Cl)nc1O CCCCCC(C)(C)C(=O)NC1CC1CNC(c1cnn2ccc(C)cc12)=O Cc1cc(C(=O)NC(C)CC(C)NC(C23CC(C2)C3)=O)ccc1Cl n1(CCn2cc(C3(C(N4CCCN5CCCC45)=O)CC3)nn2)cnc2ccccc12 N1(C(c2n(CC#C)cnn2)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)CC1 C(=O)(C#CC(=O)O)N(CCC(N)Cc1ccccc1)C1CC1 c1(C(=O)NC(C)C(C)NC(c2ccc(F)s2)=O)cc2ccc(O)cc2[nH]1 c1(C(=O)NCCNC(Cc2cccc(C)c2Cl)=O)cc2cccnc2s1 C(=O)(C(C)CS(C)(=O)=O)N1CCC(O)(CCNC(c2cncc(C#C)c2)=O)C1 C1(C)(CNC(Cc2c(C)occ2)=O)CCC(NC(c2conc2C)=O)CC1 c1(CC(=O)OC)ccc(O)c(C(=O)NC(C)CNC(=O)C(C)P(C)(C)=O)c1 C12(NC(C(C3CC3)SC)=O)CC(C1)N(C(C1CCN(Cc3ccccc3)C1)=O)C2 c1(C(=O)NC2CC(C)(NC(=O)CCC3CCCO3)C2)coc2c1C(O)CCC2 N1(C(c2c(OC)scc2)=O)CC2(C(=O)N(C3CCCOC3)C)CCC1CC2 C1(CNC(c2cc(C)c(Cl)s2)=O)CCN(C(=O)CCSCC(N)=O)CC1C C(C(N=c1[nH]c(Cl)ncc1C1CC1)C(C)C)NC(COc1ccc(C)c(C)c1)=O N1(C(Cc2cc(C)sc2)=O)CCC(C)CC1CNC(c1coc(C2CC2)n1)=O C1(C(=O)NC2C3CN(C(CC(COC)(C)C)=O)C2CC3)CSc2ccccc2O1 CC(CC(=O)NCCN(C(c1cnn2c1NCC(C)C2)=O)CC)C(F)(F)C(F)(F)F Cn1cnc2nc(=NCCN3CCCC3)[nH]c(NC3C(NS(=O)(=O)C(F)F)C3)c12 C1(CNC(CNS(C)(=O)=O)=O)CCC12CCN(C(c1c[nH]c(C(N)=O)c1)=O)CC2 Cc1cccnc1CCC(=O)NCC1COCCO1 C(=O)(NNC(=O)c1ncccn1)NC.c1(C(C)OC(C)(C)C)ccc(O)cc1 N1(C(C(CC)N(C)C)=O)CCCC(CO)(NC(=O)COc2cccc(Cl)c2)C1 Cn1cnc2nc(N3CCC(C(C)(C)C)(CNC(C4CC=CCC4)=O)C3)ncc12 C1(C2CCC2)(C(N2CCCC(NC(c3n(CC)ncc3Cl)=O)C2)=O)CCC1 CC1(C)CC(NC(=O)CC(O)C2CCCC2)CN1C(=O)CCSC1CCCC1 Cc1cn2cccc(C(=O)N(C3CCN(C(=O)CC(O)CC(C)(C)C)C3)C)c2n1 C(N=c1ncc(I)c[nH]1)C1OCC(CNC(Cc2cc(C)on2)=O)C1 N1(C(c2nc(C)n(C)c2)=O)CCC(O)C(N(C(=O)CC2CC(F)C2)C)C1 C1(C2CCOCC2)(NC(C(CSC)C)=O)CCN(C(=O)COCC(C)(C)C)C1 C(=O)(C1CCc2cccnc21)NCC1(C)C(C)CN(C(c2c(C)c[nH]n2)=O)C1 CN1CCC(C(N2CCC2C2CCC2)=O)(NC(C2CSCC(=O)N2)=O)C1 N1(C(C2CC(C3CC3)=NO2)=O)CCN(C(C2CCC3(CC2)CC3)=O)C2(CC2)C1 C1(C(C)(C)NC(C=CC)=O)CCN(C(C2CCC(c3ccccc3)O2)=O)CC1 c1(CC)ncsc1C(=O)NCCC1CC(NC(C2(C)CC2Br)=O)C1 c1(C(=O)NC(CC2CN(C(CSCC)=O)C2)C)ccn2ncccc12 N1(C(CC(CCC)C)=O)CCC(C2CCN(C(c3cnnc(C4CC4)c3)=O)C2)C1 N#Cc1cnc(NC2CCC3CN(C(c4ncccn4)=O)CC23)c(Br)c1 C1(C(N(C(C)(C)C)CCO)=O)CCCN(CCCNC(c2cn(C)nc2)=O)C1 Cc1ccc(C)n1CCC(=O)NC1(CO)CCN(C(c2cnc(C(C)C)[nH]2)=O)C1 CON(C)CC(O)Cn1cc(NC(=O)CC(c2cccs2)NC(N)=O)cn1 C(=O)(C1=Cc2ccccc2C1O)NC(CC1CN(C(CNS(CC)(=O)=O)=O)C1)C c1(C(C)COC(=O)CCOCCO)ccccc1F C(=O)(CCCCC(N)=O)NC1CN(C(c2cc(OCC)n[nH]2)=O)CC(C)C1 C(=O)(CC(C)C(F)(F)F)N1C(CC)C(NC(=O)C2=CCCCC2)CC1 c1(C(N2C(C=CC(NOCC(=O)OCC)=O)CCC2)=O)cnnc(C)c1C Cc1ccc(C(=O)NCCN(CC(=O)NC2C(c3cn[nH]c3)C2)CC(C)C)cc1C c1(C(=O)NCC2(CNC(C(C=C)(C)CC)=O)CC23CCC3)ccsc1S(C)(=O)=O C1(NC(c2c(CC)ccs2)=O)CCC2CC1CN2C(c1oc(C)cc1C)=O C1(NC(C2N(C(C3N(CC)CCC3)=O)CC3CC32)=O)CC2COCC(C1)C2 N1(C(C(CSC)OC)=O)CC(C(=O)NC(c2csc(C)n2)C)C2(CC2)C1 C(CCCC(C)(C)C(=O)NNC(=O)c1ccoc1Cl)NC(C1C(C)OCC1)=O c1(OC)cc(C(=O)NC2CN(C(=O)CN3CCC3C)C2)c(C(F)F)cc1OC C1(CNC(CC2CC(=C)C2)=O)CC2(CC2)CN1C(c1cccc(SC)c1)=O N1(C(c2c(OC)cccc2)=O)CC(C)CN(C(c2cccc(C)c2N)=O)C(C)C1 C1(C(N(C(C)(C(N2CCC(O)(CO)C2)=O)C2CC2)C)=O)CCC(F)(F)CC1 c1(NC(C2C3CN(C(CSC(C)C)=O)CC32)=O)cc(F)ccc1C(F)(F)F N1(C(c2csc(C)c2C)=O)CCCCCC1C(=O)Nc1cccc(C#N)c1 O=C(C1=CC2(CCOC2)C1)N1CCCC(CCNC(C2(CO)CC2)=O)C1 c1(C(N2CC(C=C)OCC2)=O)ccc2c(n1)CN(C(=O)C(N)=O)CC2 c1(C(N2CC3=C(CN(C(C(CCC)C)=O)C3)C2)=O)cc(F)c(F)c(F)c1N C1(C(C)NC(=O)CCN(C)C)CN(C(=O)CC2CCCN(C)C2)CCO1 Clc1cccc2ccc(CN3CCCN(c4nccs4)CC3)nc12 C(CCC1CC1)(C(=O)NCc1ccnn1C)NC(c1cc(C(C)C)[nH]n1)=O Cc1cc(C(=O)NC(C2CCCN2C(=O)Cc2n[nH]c(=N)s2)C)ncc1F c1(CC(=O)NCCC2N(C(C3C(C)(C)CCC3)=O)CCC2)c(F)cccc1F c1(N2CCCC(C)(CC)C2)nc2ccsc2c(=NC2C3CCCCC23)[nH]1 c1(C(N(C(C)CCNC(c2nsnc2O)=O)C)=O)cscc1S(C)(=O)=O C1(O)(C(N2CC(O)(C(C)NC(c3nc(C)nn3C)=O)C2)=O)CC2(CCOCC2)C1 C(=O)(C1=CCN(C)C1)N1CC=CC(NC(C(C)(C)N(C)C)=O)C1 C1(CN(C(COC(C)C)=O)C)COCCN1C(=O)CC12CCCC1C2 C(CC(C(=O)NCCc1cscn1)NC(=O)Cc1cnco1)=CC C1(CNC(C=CCC)=O)C(CC)CCN1C(=O)C(CCC)N(C)C c1(C(N2CC(CNC(C=CCOC)=O)C(C)C2)=O)cc2cc(F)ccc2[nH]c1=O c1(CN(CC(C)NC(C2(C)CCNC2=O)=O)C)ccc2ccccc2c1 c1(C(=O)NC2C(NC(CSC)=O)CCCC2)c(C)nn(C)c1F C(c1cn(C)c2ccccc12)=CC(=O)NC1CC(NC(C(CO)N(C)C)=O)C1 c1(C(C(=O)NC2CCCC2)N(C2CCC2)CC)ccc(OC(C)=O)c(F)c1 CCCC(C#N)C(=O)N1CC(OC)C(NC(C2CN(C)C2)=O)C1 C(CN=C(NC1CCC1)N1CCCC(C)C1)C1CCN(C(C)=O)CC1.CC#N N1(C(CCc2ccc(C)c(C)c2)=O)CC(NC(C2CC=CCO2)=O)CC12CCC2 C1(CCCCC)CCC(C(=O)N(CCCNC(=O)C(C2CC2)SC)C)O1 n1(CC(N2CC(F)(CNC(C3(COC)CC=CC3)=O)C2)=O)ccc(=O)c(O)c1C c1(C(N2CCCC(CNC(c3cncc(C)c3Cl)=O)C2)=O)cc2n(c1)CCSC2 Cc1cc(CSCOc2nnnn2C2CCCOC2)co1 C1(CC(=O)NCC(C(=O)NC)C)CC2(C1)CN(C(=O)NC1(O)CCCCCC1)C2 C1(C(=O)NCCCCNC(c2scc(C)c2C)=O)C2CCC(C2)C1(C)C C1(C(=O)NC(COC)C(=O)N2CC(N3CCOC3=O)C2)(CC)CNC(=O)C1 C1(CC#C)(C(N2CCC(O)(CCNC(c3ccc(O)nn3)=O)C2)=O)CCCCC1 CN(CC(F)(F)F)NC(=O)C1(c2ccc(F)cc2)CC1(Cl)Cl c1(C(N2CCN(C)C(CO)C2)C(=O)NC(C(=O)OC)C)ccc(Cl)c(Cl)c1C C12(C(N(CCN(C(=O)C=C3CCCC3)CC)CC)=O)CCCC1OCC2 C1(NC(C2N(CC#C)CCC2)=O)CN(C(C2(CO)CC2)=O)CC2(CC2)C1 C(=O)(C(O)CC[S+](C)C)N1CCCC(O)(CNC(CCN(C)CCO)=O)C1 C(C1=CCSC1)(c1nnnn1CCN1CCOCC1)NC(C)(C)CCO c1(C(=O)NCC2N(C(CCC(C)OC)=O)CC3CC32)ccc2c(c1)CCCO2 N1(N(CCC(N2CC(C(=O)OC)C(C)(C)C2)=O)CC)C2CCC1CC(C)C2 C1(C(=O)NC2(C)CCCC2NC(=O)C(O)Cn2cncn2)CC2(CCC2=O)C1 C1(CC(=O)N(C2CCN(C(=O)CN(C)C(=O)C3CC3)C2)CCC)COC(C)(C)C1 N#CC1(C(F)(F)F)CC1CC(N1CCC1CNC(=O)COC(F)(F)F)=O c1(OC)cc(N)c(C(=O)NCC2CC2NC(=O)Cc2ccccc2)cc1Br N1(C(CCCNC(C(CCCC)(C)F)=O)=O)CCCC2(CCCC2)C1 C1(CCNC(CSC(C)(C)C)=O)CCN(C(C2(C(NS(N)(=O)=O)=O)CC2)=O)CC1 c1(C(=O)NCC2CCCN(C(C(CC)=CCCC)=O)C2)cc(F)ccc1C1CC1 C(CC(C)(C)C(c1nnnn1C1CC1)NC1(CF)COC1)OC Cc1cnc(C(N2CC(F)CC2CNC(C2CSCN2C(=O)C(C)C)=O)=O)cn1 C1(CCC#C)CCN(C(=O)CC2(CNc3ccsc3)CC2)C1 C1(CNC(C=CCCC=C(C)C)=O)CN(C(=O)Cc2ccns2)CCC1(F)F N1(C(COC(C)C)=O)CCCC(N2CCN(C(c3c[nH]nc3F)=O)CC2)C1 C1(C(N2CCC(C)(CNC(CCC=C(C)C)=O)C2)=O)CN2CCCC2CO1 Cc1ccc(C(N2CC(CNC(c3cc(C)sc3C)=O)CC2C)=O)cc1O C1(C(=O)NCC2CCN(C(C3CCC(C)S3)=O)C2)CCC(Cc2ccccc2)CC1 C1(NC(c2cc(C)no2)=O)C2CCCN(C(=O)C(F)CC3CCOC3)C2C1(C)C c1(CC(=O)NCC(C2CCC2)NC(=O)COC(F)F)cccc2ccccc12 C(=O)(C(C)(C)C(O)C(C)C)N(CC(CC)NC(=O)CCC(C)(C)[N+](=O)[O-])C CCC(CC)CCC(=O)N1CCN(Cc2cnc(N3CCOCC3)nc2)CC1C N1(CC)N=C(C(=O)NCC23CC2CN(C(=O)CC2CCC24CCC4)C3)CCC1=O c1(OC)ccc(C(=O)NCC2CC(NC(=O)COc3ccccc3O)C2)cc1F C(=O)(CCCC(=O)N1CCCC(CCC(=O)NC(CCO)C(F)(F)F)C1)OC C1(N(C(CCCCSC)=O)C)CC2CCC(C1)N2C(c1cnc(O)cc1C)=O S(=O)(=O)(c1cnc(N2CCOCC3(CCOCC3)C2)c(Cl)c1)NCCS(C)(=O)=O N1(C(c2c(C)scn2)=O)CCC(CNC(C2CCC(NC(N)=O)CC2)=O)CC1 c1(OCC)ccc(CC(c2ccccc2)C)cc1.N12CCOCC1CNC(=O)C2 N1(C(C(c2cccc(F)c2)(C)O)=O)C2CCC1CN(C(=O)C1=CS(=O)CCC1)C2 CC1(C(=O)NCC(CNC(=O)Cc2cccc(O)c2)CO)CCCNC1=O C1(CNC(c2cc(Cl)ccn2)=O)CCN(C(=O)CCCc2cccs2)CC1 c1(OC)ccc(C)c(C(c2nnnn2C2COC2)NC2CCCCCC2)n1 n1(CC(=O)NC2CCC(NC(C(CC=C)NC(C)=O)=O)C2)ncc(C)cc1=O C12(C(=O)OC)CC(C1)C(NC(N1CCCC1)=O)CCS2.C123CC(C1)(C2)N3 C1(C(N2CCC(C(C(=O)NCc3c(C)n[nH]c3C)C)C2)=O)CC12CCOCC2 O=C(C(CO)C(F)(F)F)NCC1CCN1C(c1cnccc1C1CC1)=O C1(CC(=O)N(C(C)C)CCN(C)C)CN(C(C2CC2(Cl)Cl)=O)CC1C N1(C(C2CCN(C(C3C(C)(C(F)F)C3)=O)CC2)=O)CCC2(C=CCO2)C1 C12(NC(=O)C3CC3)CCN(C(=O)CCc3cc(Br)cs3)CC1C2 Cc1c(Cl)ccc2cc(C(=O)NCC(CO)NC(=O)COCC(C)C)cnc12 c1(C(N(C(CNC(C2C(C3C(C)C3)C2)=O)C)C)=O)ccnc2cc[nH]c12 CN1CC(O)CC1(C)C(=O)NCC(C1CCCC1)NC(C1CC2(C1)CC(C)C2)=O C1(C#N)(NC(C(c2ncn(C)c2)O)=O)C2CC(F)(F)CC2C1 c1(C(=O)NCCC(=C)CNC(=O)CSCCCC)ccccc1CC C(CCCC(=O)N(CC(=O)NC(c1nn[nH]n1)C)CC1CC1)(OC)OC CC1(C)OC2(CNC(C3CCCCS3)=O)CC1(NC(C1CC(CF)C1)=O)C2 C1(NC(c2csc(CO)n2)=O)CCCCN(Cc2ccccn2)C1 N1(C(CCN(C(=O)COC2CCCCC2)CC)=O)CCN2C(=O)CCC2C1 CON1CCC(CC(=O)NC(C)CN(C(=O)CSC)CC2CCOC2=O)CC1 C1(C(=O)NCC(CC=C)NC(=O)C(C)NC(=O)CC)(CO)CCCCC1 c1(C(N2CC(OC)C(NC(c3cnc(C4CC4)s3)=O)C2)=O)ccc(F)c(C)c1 N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(=O)C(C)(C)OC)CC1C CCC(C)C(=O)NCC(C1(O)CN(C(=O)CSCc2ccccn2)C1)(C)C CC1=NNC(=O)C1CC(=O)N(C)CC1CN(C(=O)C(F)=C2CCC2)C1 C1(CNC(C2C(C)C2)=O)CCN(C(=O)CN2CCS(=O)CC2)CC1 CN1CCCC1CC(=O)N(C(C)(C(=O)NC(c1nc[nH]n1)CO)C1CC1)C N1(C(c2c(CC)cccc2)=O)CCCCCCC1C(=O)Nc1ccc(OC)cc1C c1(C(C)=O)cnc(C)c(SC2CC3CC2CO3)c1 N1(C(c2c(C)ocn2)=O)CCC(c2nnc(CNC(c3cnc(O)o3)=O)s2)CC1 c1(C(N2CC(NC(C3(F)CCCN(C)C3)=O)CC2(C)C)=O)cccc2nn[nH]c12 Cc1ccc(=O)n(CC(=O)NCCNC(=O)C(O)CN2CCOCC2)n1 C1(NC(c2c(CNC(c3ocnc3C3CC3)=O)n[nH]c2)=O)CCOCC1F c1(C(=O)NC2(CF)CCN(C(c3cnn4ccsc34)=O)C2)ccc(Cl)c(O)c1 C(=O)(C(C)(C)CC(C)C)N(CCCNC(c1ccc(-c2csc(C)n2)cc1)=O)CC C12(C(N3CCCC(NC(c4ccnc(C)c4N)=O)C3)=O)CCCCN1CCC2 C1(NC(CC2C(NC(c3c(C)ccnc3O)=O)CC2O)=O)CCN(C)CC1(C)C CC(CCC(C)(C)C)C(=O)NCC1CCCCN(C(=O)CP(C)(C)=O)C1 C1(CC(C)C)CCCCN1C(=O)NCCCSCCCO C(CCC(C(=O)NCCn1cnccc1=O)NC(=O)Cc1cnsc1)OC CCC(CN(C)C)C(=O)NCC1CC(C(=O)NC2CC(C)(C(N)=O)C2)CO1 c1(C(N(c2ccc(C3(C)CC3)cc2)C)=O)ccc2c(c1)CCC2=O c1(C(=O)NCCC2OCCN(C(CCC)=O)C2)cnc(O)cc1O C1(C(=O)NCCC2=CCN(C(C(CC)OC)=O)CC2)Cc2cc(C)c(C)cc2O1 c1(NC2COCCN(C(c3c(OCCC)cccc3)=O)C2)ncc2c(n1)CCC2 c1(C(=O)NC2CC(CNC(C(Br)=C(C)C)=O)C2)ccc2nn(C)cc2c1 n1(CC(=O)NC2C(CNC(c3c(CC)nc[nH]3)=O)CCC2)ncc(C#N)c1N c1(C(=O)NC2CCN(C(CSC(C)C)=O)C2C)cnn2c1OCC1(CC1)C2 Cc1cc(CC(=O)NCC2CC(F)(CNC(C3(C)CC3C(F)(F)F)=O)C2)c(C)s1 C1(OC)CC(C(=O)NCC2(S(C)=O)CC2)N(C(c2ccsc2)=O)C1 N1(C(c2oc(CC)c(C)c2)=O)C(C(=O)NC2CCOC2C2CC2)CCC12CC2 c1(-c2cncc(NCc3cccc(OCC)c3)n2)ccc(F)cc1CO N1(C(COC(CC)C)=O)CCCC(n2cc(CSCC)nn2)C1 C1(C(=O)NC2C3OCC(NC(CSC)=O)(C3)C2)Cc2c[nH]cc2S1(=O)=O Cc1cccc(C2CCCN2Cc2cc(C(N3CCOCC3CO)=O)sc2Cl)n1 C1(NC(CCN(C2CC2)CC)=O)CCCCC1NC(=O)Cc1cnnn1C C1(C#N)(C(=O)NC(C)CCCNC(c2cnn(CC3CCC3)c2)=O)CC12CCC2 C=CCCCCCC(=O)NC(C1(O)CCCN(C(C2(n3cccn3)CC2)=O)C1)C C1(CNC(C2CN(C(C)=O)C2)=O)CN(C(=O)CC2(O)CCCC2)CC1C C1(C(C(CC=C(C)C)=O)=O)C2CCC1(c1cccs1)C2.C(CN(C)C=O)NC1CC1 C1(C(=O)NCC(CO)NC(C2COCCO2)=O)CC2(C1)CC1(CC1)C2 c1(-c2cn(C)nc2)ccccc1C(=O)NCCN1CCN(C(=O)CC(C)(C)O)CC1 CS(=O)(=O)c1ccc(OC(F)F)c(C(=O)Nc2ccc(N3CCCCC3)cn2)c1 c1(N(CC(Cc2ccc(F)c(F)c2)OC)C(C)=O)nc2c(C)cccc2s1 O(N=Cc1ccc2c(c1)CCO2)C(N=c1[nH]nc(CCC(=O)OC(C)(C)C)s1)=O N1(CC(N2CC(CC=C)(NC(=O)C(c3cnn(C)c3)C)C2)=O)CCS(=O)(=O)CC1 CN=c1[nH]c(SC)ncc1CN1CCC(F)(F)C(C(N2CCC2CO)=O)C1 N1(C(CCCCC#N)=O)CCCCC(n2cc(C3(O)CC3)nn2)C1 C#CCCCCC(=O)NCC1(F)CC(NC(C2COC(C)C2)=O)C1 C1(C(N2C(C(C)NC(c3ccc(N)cc3)=O)CCCC2)=O)CC2(C1)CC2(F)F CC(C(=O)NC(CNC(=O)CC1CSC1)C1CC1)OC(C)(C)C CC1C2(CCC2)CN1C(=O)C(Cn1cccn1)NC(c1ccc(C#N)cc1)=O C1(CC(=O)NC2CC(NC(c3c(OCC)cccn3)=O)C2)COC2(CCC2)CO1 C1(C(N(CCCCNC(c2c(C)ncc(C)c2)=O)C)=O)CCCCC12CCC2 N1(C(c2cc(-n3ccc(C)n3)no2)=O)CCN(C(=O)C(O)C(F)F)CC1C C1(NC(c2c(CC)ncs2)=O)CN(C(=O)Cn2nc(C)oc2=O)C2CCCC12 c1(C(N2CC(F)CC(NC(c3cc(C)[nH]n3)=O)C2)=O)ccc2c(c1)NC(=O)CS2 C1(C(=O)NCC(CC)N(C)C)C=CCN1C(=O)CCC1CCCCC1 c1(CNCC2(N(C)C)CCCC2)ccc(Cl)c(F)c1 C(=O)(C=CS(C)=O)N(C(C)CNC(=O)CNC(c1ccccn1)=O)CC N1(C(CCCC(=O)N(C)C)=O)CCC2CCCN(C(=O)COCC(F)F)C2C1 CC(C)(C)CC(C(=O)NCCC1CCOC1(C)C)NC(c1ccncn1)=O C(=O)(CCCC(=O)N(C(C1CCN(C(=O)C(F)(F)CO)C1)C)CC)OC N1(C(C2(CC(C)=O)CCC2)=O)C2CCC1CC(NC(=O)C(C)N(C)C)C2 C(C(C)(O)C(=O)N1CCC(C(C)CNC(c2ccoc2C2CC2)=O)CC1)OC c1(N2C3CC(NCC4CCCN(C(C)=O)C4)CC2CC3)ncnc2scc(Br)c12 C1(CC(=O)NCC(C)(C2CC2)NC(C(C)Sc2ccccn2)=O)CCC(O)CC1 N1(C(C2(COCC)CC2)=O)CCCC(n2cc(C3(C4CC4)CC3)nn2)CC1 C=CCC(CC)C(=O)NCCCNC(=O)CCCc1ccc(Br)c(F)c1 N1(C(CC2CCCC(C)C2)=O)CC2(C)CC1(C(=O)NC(C)CN1CCCC1)C2 N1(C(c2c(C)c[nH]c2)=O)CCC(CO)C(NC(c2nc(C)c(C)s2)=O)C1 C1(F)(C(=O)NC(CC)CCOC)CCN(C(=O)C(C)(C)CCF)CC1 C1(CNC(=O)NC2CC(OC)C2)(Cc2cccc(Cl)c2)CCCCCC1 CC1C(NC(=O)C=CCN2CCOCC2)CCCN1C(c1cnn[nH]1)=O N1(C(CC(CC=C)NC(=O)CCC(F)(F)F)=O)CCc2cccc(C)c21 CCCCC(C(=O)NC(CNC(=O)Cn1ccc(C(=O)OC)n1)C1CC1)NCC C1(C(N(CCC)C)=O)CCN(C(=O)CN2CCC(C(C)O)C2)C1 C1(C)(CC(=O)NCCC(C)N(C(=O)C(Cl)=CCl)C)CC(F)(F)C1 n1(C(C)C)ncc(F)c1C(=O)NCC(C)CNC(=O)C(C(C)C)N1CCCCC1 c1(C(N2C(C)(CNC(c3cnc(O)o3)=O)CCC2)=O)cc(F)c(Cl)cc1Cl C1(NC(c2[nH]c(=NCC)sc2)=O)CCN(C(=O)C(C)OC2CCCC2)CC1(C)C c1(NCc2occ(C)c2)nc(C)cc(=NC2CCS(=O)(=O)C(C)C2)[nH]1 N1(C(c2occ(C)c2)=O)CCC(C(=O)NCCC2CCC(C)(C)C2)(CF)C1 Cn1nc2c(c1N)CN(C(=O)C(C)(C)CC(C)(C)C)CC2 C1(CNC(CCC(=C)Cl)=O)CCN(C(c2ccncc2Cl)=O)C12CC2 C(CCC(=O)N1CCCC1C(C)(C)Cn1cc(C(C)(C)C(C)C)nn1)OC CC(O)CC(=O)N(C(c1ccccc1)CNC(=O)C(C)(C)c1nncn1C)C c1(C(=O)NCC(CC(C)C)NC(=O)C2=COCCC2)cc2c(s1)CCSC2 C1(NC(c2cncn2C2CC2)=O)CN(C(C2OC3CCC2C3)=O)CC1C(F)F Cc1cccc(NC(=O)CCC2CCCN2c2cc(C#N)ncn2)c1F C123CC1CC1CN(C2)C(=O)C1(C1CC1)CC(=O)CC(=C)CC(C)CNC3=O N1(C(C=CC(=O)NC)=O)CCC(C)C(NC(=O)CC2C=CCC2)C1C n1(CC)cc(S(=O)(=O)NC2CCCC(C(=O)Nc3cnc(Cl)c(F)c3)C2)cn1 C12(C(N3CCC(c4ccccc4Cl)(OC)C3)=O)CC1COC2(C)C c1(CC(=O)NCCC2CCSCC2)c[nH]c2cccnc12 c1(C(N2CCOCC(NC(C3CCCCC3(F)F)=O)C2)=O)ccc2ccsc2c1 c1(N2CCCC(CC#N)C2)ccc(C(F)(F)F)cc1S(=O)(=O)NCCSC(F)F n1(CCCC(=O)NC(c2cn(CC(C(=O)OCC)O)nn2)C)c(O)nnc1O CC1=NOC(C)(CNC(C2CCC(NC(=O)C(C)(C)C3(O)CCC3)CC2)=O)C1 Cc1ccc(NC(=O)C(C2CCN(C(c3cncn3C(C)C)=O)CC2)C)c(C)n1 C1(C(=O)NCC2CC(NC(c3cnn(CCO)c3N)=O)C2)(OC)CS(=O)(=O)C1 c1(C(N2CCN(CCC#N)CC2)C(=O)NC)ccc(Cl)cc1C c1(CC(N2CC(NC(c3nnn(CC)c3C)=O)(CO)C2)=O)c(C)nn(C)c1Cl c1(CC(=O)NCC2CC2NC(C2CCc3nc[nH]c3C2)=O)ccc2c(c1)CCC2 C1(C(N2C(CNC(=O)CO)CC(F)(F)C2)=O)CCn2c(C(F)(F)F)nnc2C1 c1(Sc2ncc[nH]2)cc(N2CCOCC2)ncn1.C12CC(C1)NC2=O N1(C(C(C)NC(CC)=O)=O)CCC2C(CCCN2C(C2SCC=C2C)=O)C1 C1(NC(C(C)OCCC#C)=O)(CNC(c2snnc2C)=O)CCOCC1 c1(C(N2CCC(N(C(COCCOC)=O)C)CC2)=O)cc(F)cc2ccncc12 N1(C(CN(C(=O)CCn2cc(Cl)cn2)C)=O)CCN(C(=O)Cc2ncon2)CC1 c1(C(=O)NCC(N(C(C(=Cc2cccs2)C)=O)C)C2CC2)ncccc1C C(C(N=[N+]=[N-])C(=O)N1CCC(CN(C(=O)CCCCCOC)C)CC1)OCC N1(C(c2cccc(C)c2)=O)CCC(F)(CNC(=O)Cc2cncnc2O)CC1 CC1C(NC(c2cnoc2C2CC2)=O)CC2CCC1N2C(C1CCC(F)C1)=O C(=O)(C(CC(F)F)NC(c1csc(O)n1)=O)NC(c1cncs1)C C1(C(C)C)CN(C(=O)C=Cc2cccs2)CCN1C(=O)CSCC1CCCCO1 N1(C(c2cccc(C(=O)OC)n2)=O)CCN(Cc2ccc(I)c(F)c2)CC1C#N N1(C(C23CC(CC)(C2)C3)=O)CCCN(Cc2nc(Cl)sc2Cl)CC1 c1(C(=O)Nc2[nH]c(=NCc3cc(OC)c(Br)cc3)sc2)ncnc2c1CCCC2 Fc1ccc(Nc2ccc(-c3nc[nH]n3)cc2)c(C(F)F)c1F N1(C(c2cnc(C(C)(F)F)s2)=O)CC(NC(c2ccc([N+](=O)[O-])o2)=O)C(C)(C)C1 c1(C(=O)NC2(CNC(c3cnn4c3OCC4)=O)CCC2)cc(F)c2cn[nH]c2c1 c1(C(=O)NC(C2CCN(C(=O)C(C)(C)C)C2)C)ccc2ccc(Br)cc2n1 N1(C(C2N(C(CCC(=O)NCC)=O)CC(O)CC2)=O)CCOC2C(O)CC12 C1(N(C(CC(OCC)OCC)=O)C)C2CN(C(c3cncc(OC)c3)=O)CC12 C1(NC(=O)C=CC2CC2)C2CCCCN(C(=O)CCc3ccc(Br)c(F)c3)C12 n1(CCC(N2CC3(CCCCC3)C2)=O)sc2ccccc2c1=O CN1CC2CC1CN2C(C1(F)CCN(Cc2ccc(I)cc2Br)CC1)=O c1(CC(=O)OC)csc2c(C(F)(F)F)cccc12.C1(=O)C(C(C)O)N1 C1(CC=C)(NC(C2C=C2C)=O)CCCN(C(c2sc(SC)cc2C)=O)C1 N1(C(C(C)CC2CC2)=O)CCC2CCN(C(c3cc4cccnn4c3)=O)CC12 C1(NC(C(C)O)C2CCCC2)CCN(c2cc(O)ncn2)CC1 C1(C(=O)OC)CCCCC1S(=O)(=O)Nc1ccc2nc(C)ccc2c1 C(=O)(CCC(=O)NC(=O)NC)N1C(CN(C(CN(CC)CC)=O)C)CCC1 C12(NC(c3[nH]cc(C(=O)OC(C)(C)C)c3)=O)CCC(CC1NC(C1CC1(C)C)=O)C2 CC1CCC(C)(C(N2CC(O)(C(C)NC(=O)Cc3cccnc3O)C2)=O)C1 Cn1nnc2c(C(=O)NC(CNC(c3cc[nH]c(=N)c3)=O)C3CC3)ccnc12 C1(C(=O)NCC(O)C(C)(C)C)(CC)CCN(C(c2cccc(O)c2)=O)C1 C12(NC(C(C(C)(C)O)F)=O)CCCC1N(C(c1cc3ccsc3s1)=O)CCC2 c1(C(N2CC(CN(S(CC)(=O)=O)C(C)C(=O)OC(C)(C)C)C2)=O)ccc(O)nc1 C=CCN=C(NCC(C)C#N)NCC(Cc1ccccc1)C(F)(F)F N1(C(CCCC#C)=O)C(CNC(c2ccc(F)cn2)=O)CC2CCCC12 c1(CC)cc(C(=O)NCC2CC(NC(=O)CCSc3ccccc3)C2)c(C)o1 c1(OCCOCCOC)ccnc(N)c1.c1(OC(F)F)ccccc1OC c1(C(N(C(CCNC(CN(C(C(C)C)=O)C)=O)C)C)=O)cnn(C(C)C)c1F C#CC1(NC(=O)C(C)NC(C2C3CN(C)CC23)=O)CC2CCCC12 C(CNC(=O)CNC(C)=O)(CC(F)(F)F)NC(C(c1cccc(OC)c1)(F)F)=O N1(C(CCC)=O)CC2CC1C2NC(=O)C(O)Cc1cc(Cl)sc1Cl N1(C(C2COCC(C)O2)=O)CCC2CCCC12C(=O)Nc1ccccc1O c1(NC(C(C2CCN(C(c3ncco3)=O)CC2)C)=O)cc([N+](=O)[O-])ccc1Cl C(=O)(NNC(=O)C(=O)N1CCCCC1)C1SCC(C(=O)OC)C1 CCCC(C)C(c1nnnn1C(C)(C)C)NCc1ccc(Cl)o1 c1(C(N(C)CCOCCNC(=O)CSCCC(C)C)=O)c[nH]nc1Cl c1(CC(C)(C)C)ccccc1-n1cc(C(=O)NCCc2cnc(C)[nH]2)nn1 c1(C(=O)Nc2ccc(CC3CC3)s2)cccc(CC2C(NC(C)=O)CC2)c1 S(=O)(=O)(c1ccc(CN2CCS(=N)(=O)CC2)s1)NCc1nc(C)[nH]n1 C(c1ccc(Br)cc1)=C(C(=O)NC1CC1)N(C1CCCCC1)CCC c1(NC(C2N(C(CCN(C)C)=O)C3C(C2)C3)=O)ccc2c(c1)CCOC2 CC1CCCC=C1C(=O)Nc1c(C2CC2)cccc1Cl C1(O)(C(=O)NCC2C3CN(C(CCCCOC)=O)C2C3)CCc2ccccc2C1 C(c1ccc(Br)c(C)c1)=CC(N1CC2C(NC(COC(C)=O)=O)(CC2)C1)=O c1(C(=O)NCC2CC(OC)CN2C(=O)CC(C)C)ccn2c1CCC2 C1(NC(=O)Cc2cccs2)C2CC3CC(C2)CC1(CNC(C1CCCO1)=O)C3 c1(NC(C2(CCCC)CCCC2)=O)cccc(F)c1C.n12ccc(c1)C(=O)NCC2 CCCC(C)C(=O)N1CC(OC)CC1CNC(c1ccccc1Br)=O CONC(=O)C(=O)NCCC(=O)NCCC(C)N1CCCC1 C1(CC(=O)NC(C2(CNC(=O)C=CCN3CCCC3)CC2)C)C=CS(=O)(=O)C1 S(=O)(=O)(c1ccc(NC2C=CCCC2)cc1Br)N1CCC2CCN(C)CC2C1 N1(C(CN(C2CCSC2)C)=O)CCN(C(C2(C)CC(OC)CN2C)=O)C2(CC2)C1 C1(NC(=O)NC2CC(Cn3cccn3)C2)CC(C)(CC(C)C(C)(C)C)C1 CC1(C)CC(C(N2CC3(C2)CN(C(=O)C=Cc2ccccc2Cl)C3)=O)C(C)(C)O1 Cc1cccc2c(C(=O)NC(C)(CNC(c3ccc(O)cc3)=O)C(C)C)csc12 c1(C(N2CCC(CCC(N3C(C)(CCC)CCC3)=O)C2)=O)cc(O)nc(C)n1 C12(NC(C(C(C)C)Nc3cc(=O)n(C)c(O)n3)C3CC3)CC3CC(C(=O)N1)C2C3 CC1CN(C(=O)CCCC2CCCO2)CC(C(=O)NCCN2CCNC2=O)O1 c1(C(N2CC3C(CNC(C(CCCC)CC)=O)(C3)C2)=O)cccc2oc(=N)[nH]c12 c1(C(=O)NC2(CC(=O)Nc3ccnnc3)CCC2)ccc(Br)c(C(F)(F)F)c1 N1(C(C(C)OC)=O)CCCCC1C1CCN(C(=O)C(C)C#N)C1 c1(C(=O)NCC2CN(C(c3c(CC)ocn3)=O)C3C2C3)ccc(C(F)F)c(F)c1 c1(CCC(=O)NC2C(NC(C=Cc3ccc(C)o3)=O)CC2)c[nH]c2ccccc12 C1(C(=O)NC(CCOCC)C(=O)NCC2CCSC2)CC2CCCC2C1 C1(CNC(CS(CC)=O)=O)CC(C(C)C)CCN1C(=O)Cc1cccnc1 CS(=O)(=O)c1cc(C(=O)NC2CCC(CNC(c3ccoc3)=O)CC2)co1 c1(OC)ccnc(C(N2CCCC(CCNC(C3C(C)C3C)=O)C2)=O)c1F c1(C(C(N2CC(C(=O)O)(OCC)C2)=O)C)cccc(Cl)c1 c1(C(N2CCC(C(C(=O)N(CCCC)CCOC)C)C2)=O)ccnc2cc[nH]c12 CC1C(C(=O)N2CCC(NC(C3(S(N)(=O)=O)CC3)=O)C(F)C2)=Cc2ccccc21 c1(C(N2CC3(CN(C(C(CC)(CC)CO)=O)C3)C2)=O)cc(N)c2ccccc2n1 C(=O)(CCN(OC)C(=O)c1cc(Cl)n(C)n1)N1CCC(CCC)C1 C1(CNC(C2C(COC)(CC)C2)=O)COC(CNC(c2csc(O)n2)=O)C1 C1(CNC(N(c2cn(C(C)(C)C)cn2)CCC)=O)CC2CC(OC)C2C1 N1(C(C(CCNC(=O)C=Cc2ccsc2)OC)=O)CC2COCC2(C)C1 N1(C(c2cc(CCNC(C(n3ccc(C)n3)C)=O)on2)=O)CCC(C)(CCO)C1 c1(C(N(C)CC2(O)CN(C(C=C(C)C)=O)C2)=O)cccc2c(O)ncnc12 C1(C(C)C)CN(C(=O)C(Cc2ccsc2)NC=O)CCC1NC(c1ccno1)=O N1(C(C2OCCN(C)C2)=O)CCCN(CCNC(=O)C(=O)NCCC(N)=O)CC1 C1(NC(c2ccc(CC)[nH]2)=O)CN(C(=O)Cc2sc(SCC)nc2C)CC1OC C(CC)(CC)(CCNC(c1cnc(C2CC2)[nH]1)=O)NC(c1onc(CC)c1C)=O Cc1ncc(C(=O)NCC=CC(=O)NCCCC2CC2C)s1 N1(C(C=NOC)=O)CCC(NC(C2CC(C)=NO2)=O)C2CC12 C1(NC(CCCC#C)=O)(CO)CCCN(C(c2cc3c([nH]2)CCC3)=O)C1 C12(C(=O)NC3CN(C(=O)COc4ccsn4)CC3F)CCCC(CCC1)C2O CC1CN(C(=O)CSc2ccccn2)CCCN1C(=O)CC1CCCC(F)(F)C1 CCCC(CNC(c1ccn(C)c(=O)c1)=O)C(=O)Nc1cccc(Cl)c1O c1(C(=O)OC)cnccc1C(=O)N(C(CC)C(=O)NC1(C)CC(CO)C1)C C1(NC(c2cn(CC)nn2)=O)CN(C(C2CCCCS2(=O)=O)=O)CCC1F C=CCC(C(=O)NCC(F)(C(=O)Nc1ccc(CO)nc1)C(C)C)C(C)C C(C(CO)C(C)C)NC(C(c1cn(C)nn1)NC(CCC=CC)=O)=O C(CC(CNC(c1ccnn1CCF)=O)NC(C1OCC1(C)C)=O)OC Cc1cc(C(=O)NC2CCCCC2CNC(C2CC2(C)C)=O)ccc1F CN1CCN(C(C2(C(F)(F)F)CCCCO2)=O)CC1CNC(c1cncs1)=O c1(C(=O)NCC(CNC(C2(C(C)(F)F)CC2)=O)F)cnccc1Br c1(SC)nc(Cl)c(CN2CCC3(CC3C(=O)Nc3cnc(Cl)nc3Cl)C2)c(Cl)n1 C1(NC(C2CC(=C)C2)=O)CC2(CCC(NC(C34CCC(C3)OC4C)=O)OC2)C1 C#CC1(C(N2CC(C)(NC(C3(C(F)(F)F)CC(C)(C)C3)=O)C2)=O)CCCC1 c1(Cc2ccc(C(C)(C)C)s2)ccccc1CO.C12CCN1C2=O CCC(CC)C(C(=O)NC1CCC(C(N2CCCCC2COC)=O)C1)OC Cc1cnc(C(=O)NCC2CN(C(=O)CC3CCN(C)CC3)CCC2C)c(C)c1 n1(CCOC)cc(C(=O)NC2(C)CCC(NC(=O)CC3CC3)CC2)ccc1=O CCCCCCC(CC)C(=O)NCC1(O)CN(C(c2ccnn2C)=O)C1 C(=O)(CCS(N)(=O)=O)N1CC(C)C(CNC(=O)CN2CCN(C)C(=O)C2)C1 Cc1cccc(C2(CNCC3CCCO3)CCCCC2)c1 C1(C(=O)NC2CN(C(CCc3nc(C)c(C)o3)=O)C2)CCCC2(CCOC2)O1 C(C1=CN(C(=O)NCCOc2ccc(COC(C)(C)C)cc2)CC1)OCC c1(OCC)cc(N2CC(O)(C(C)NC(c3cc(C)ncc3Cl)=O)C2)nc(C)n1 N=c1[nH][nH]c(=NC(=O)N(C2(C(=O)N(c3ccccc3)CC3CC3)CC2)CCO)s1 c1(CN(C(C(n2cc(-c3ccc(C)cc3)nn2)C)=O)C)ccc(F)c(C)c1 C1(NC(=O)COCC2CC2)CC(F)CN(C(C2C(F)(F)C23CC3)=O)C1 C(CC(C(=O)NCc1ncoc1C1CC1)NC(=O)Cn1ncccc1=O)N(C)C N1(C(CCC(=O)OC)=O)CCC2CCN(C(c3cc(OC)c(Br)s3)=O)C2C1 N1(C(C(COC)COC)=O)CCCC(N(C)C(c2cccn2C)=O)CC1 N1(C(c2cc(C(C)C)on2)=O)CCC(F)(F)C(NCc2cc(Cl)ccn2)C1 N1(C(=O)Cn2ncc(O)nc2=O)CCC2CCCC(C1)N2C(=O)C1=NOCC1 N1(C(c2cncc(CNC(C3(F)CCC3)=O)c2)=O)Cc2ccccc2C1 C(C1=CCN(C(=O)CCc2ccc(Br)s2)CC1)NC(c1cc(C)c(C)[nH]1)=O O=C(C1=CC2CCCCCC12)Nc1ccc(S(=O)(=O)NC2CC=CC2)c(Cl)c1 Cc1nc(CC(=O)NCCCC(C)NC(=O)CC(C2CC2)C2CC2)sc1C c1(NC(C2C(C(=O)Nc3n(C)nnc3)C2)=O)ccc2c(O)nc(O)nc2c1 Cc1nccc(CNC(=O)CCn2cc(C3CCOC3)nn2)c1C c1(-c2ccc(C(=O)NCc3nccn3C)cc2)cnc(CC)cc1C C(=O)(C1=COCCO1)N1CCC(NC(C(C)OCCCC)=O)(CF)C1 C1(C(=O)NCc2[nH]n(C)c(=O)n2)CCN(C(=O)C=CCN2CCCC2)C1(C)C N1(C(c2ccc(C(N)=O)s2)C(=O)NC)CCN(C)C(c2ncc[nH]2)C1 N1(C(c2cc(CC)nc(O)c2)=O)CCN(C(C2CCC(=O)O2)=O)C2CCC12 Cc1ccc(NC(=O)CCC2CCCN2C(=O)CC2CC=CCC2)c(C)c1 c1(C(=O)NCC23OCC(NC(c4c(C)nn(C)c4)=O)(C2)C3)ccc2c(c1)CCO2 c1(C(=O)NC(C(=O)N(C)Cc2cc(OC)no2)C2(C)CC2)scc(C)c1C N1(C(C(C)C)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1c1ccncc1 N1(C(CN(CCC)C)=O)CCCC(C)C1CCNC(=O)CC1CCN(C)CC1 N1(C(C2(CNC(C3CCN(C)CC3)=O)CC(=C)C2)=O)CCCC(C)C1CCC N1(C(c2cc(C)ns2)=O)CCCC(c2cn(CC(C)(C)C(C)O)nn2)C1 CN1CCCC(CC(=O)NCC(C2CC2)NC(=O)CCc2cn[nH]c2)C1 CC1CN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC1NC(c1coc(Br)n1)=O C1(NC(=O)C2CC2)CN(C(c2cnc(C3CCC3)s2)=O)CC2(CCOCC2)C1 N1(C(C2(CC=C)CCN(C(C3CC(OC)C3)=O)C2)=O)CCc2c[nH]nc2C1 C1(NC(C(F)=CCC)=O)CN(C(c2coc(C3CCOCC3)n2)=O)CC1(C)C C1(CNC(C2(C)CC(F)C2)=O)CN(C(C2CCCO2)=O)CCC12CCOC2 c1(C(N2CCN(C(CCCOCCC)=O)CC2C)=O)ccc2c(c1)C(C)CN2 C1(C2CCCN(C(C3(CO)CC3)=O)C2)(NC(c2ccnc(C3CC3)n2)=O)CC1 c1(C(=O)NC2C(N(C)C(c3ncccc3O)=O)CCCC2)coc2ccccc12 Cc1cccc(OCCS(Cn2cc(COC(C3CC4CCC3O4)=O)nn2)(=O)=O)c1 c1(C(=O)NC2CN(C(c3c(C)nns3)=O)CC3C2C3)c(N)cccc1[N+](=O)[O-] CSC=CC(=O)NC(C)(CNC(=O)C=Cc1ccoc1)CC N1(C(C(C)C2CCCC2)=O)CCC2CCN(C(=O)CC3(O)CCC3)C2C1 C1(C(=O)NCCN(C(COCCCCC)=O)CC)CC2(C1)C(F)(F)C21CCC1 N1(C(c2c(SCCC)cccc2)=O)CCC(NC(=O)CC#N)C(C)C1 c1(CC)nccn1CC(C)NC(c1ccc(Cl)s1)c1nnnn1C1(C)CC1 c1(NC(=O)NC(=O)C2CC2)cccc(NCc2ccccc2-c2cccnc2)c1 N(C(=NCC(C)C)NCC1(C)CC2(C1)CC(F)(F)C2)Cc1ncc(C)s1 c1(CC(N2CC(F)(F)C2)=O)csc(-c2cnn(C3CC3)c2)n1 c1(C(=O)NC2CC(C(=O)NCC#N)C2)ccc(Br)cc1 c1(C(N2CC(NC(COCC)=O)C2)=O)oc2ccc(F)cc2c1-c1ccccc1 C#CC1(O)CC(C(=O)NCC(c2cccc(C)c2)NC(C2CC(F)(F)C2)=O)C1 Cc1ncc(C=CC(=O)NC(C2CCCN2C(=O)C(C)(F)F)(C)C)c(O)n1 C(=O)(C(C)CCCOC)NCC1(C)CCN(C(CN(CCC)C)=O)C1 c1(C(=O)NCC23N(C(C(C)OCOC)=O)CC(C2)C3)cn2ncnc2nc1C N1(CC(=O)NC2CCC(NC(C3CC4CC3C4)=O)C2)CCCCCC1 CC1=C(C)CC(C(=O)NOCC2(CCO)CCCC2)CC1.C12(CC1)C(=O)NC2 CN1CC(C(=O)N(C(CNC(C2COC(=O)N2)=O)C2CC2)C)CCCC1=O C1(NC(C2CCC(C(=O)OC)CC2)=O)CC(F)(F)CC1NC(C1(C(N)=O)CC1)=O Cc1nc2cc(NC(C3CNCC(C)(C)O3)=O)ccc2o1 C1(C)(CNC(C(C)c2ccsn2)=O)CCCN(C(=O)C=Cc2ccsc2)C1 C12(C(=O)NC(C(C)SCC)C)CC(CN(C(=O)CC3(CO)CC3)C1)C2 c1(N2C(=O)CN3C(CC(Cl)C3)C2=O)cc(C)oc1C.c1(COC)cccc(C)c1 C1(F)(CNC(C(C)(C)c2ccccc2)=O)CCN(C(c2ccc(=O)oc2)=O)C1 CCC1=NOC(CC(=O)NC2CC(N(C)C(c3c[nH]nc3Br)=O)C2)C1 CCC(CCC(=O)NC(C)(C)CN(C(=O)C(C)(O)Cn1ccccc1=O)C)OC c1(OC)ccc(F)c2[nH]c(CNC(c3ccccc3C(C)(F)F)=O)cc12 c1(C(=O)NCC(=C)CCNC(=O)CCNC(=O)CO)cc(CO)n(C)n1 CC(C)C(C(=O)NCC1CCC(C(=O)NOCCCCC2CC2)C1)C(C)C Cc1nc(C)n(O)c1C(=O)NC1CCN(S(C)(=O)=O)C1.C12CCC(CC1)COC2=O C1(C(N(C2CCN(C(=O)C(C)(C)CCF)C2)C)=O)CCn2nccc2C1 c1(C(N(C(C)CN(C)C(c2cc(F)c(N)cc2F)=O)C)=O)cnc2[nH]nnc2c1 n1(CC(=O)NC2CC(NC(c3c(F)ccc(CC)c3)=O)C2)cc2ncccc2n1 c1(CNCC2OCCN(c3nc(C)c(Br)cn3)C2)ccc2ncnn2c1 C1(C(N2C(CC(=O)NCCC(C(=O)OCC)C)CCC2)=O)CCC(C)=C(C)C1 c1(CN2C(C(=O)NC(c3ccsc3)C)CC2)c(O)cccc1F c1(C(=O)OC)cccc2cc(CNCCC3(C(F)(F)F)N=N3)c(=O)oc12 C1(NC(CS(C)(=O)=O)=O)CC2CC1CN2C(c1cnc(-c2ccoc2)s1)=O C1(C(N(CC(C)CNC(C2CC2c2ccsc2)=O)C)=O)CS(=O)(=O)CC(=O)N1 N1(C(C2CC(OCC)C2)=O)CC=CC1C(=O)N(CC(C)(C)CO)C CC(CC(F)F)C(=O)NCC1CCN(C(=O)CC=Cc2ccc(F)cc2)CC1O c1(C(=O)NC2CC3CC(NC(C(F)=CC)=O)CC32)cc(Br)c(F)cc1F N1(C(=O)NCc2ccn(C)n2)CCOC(c2nc[nH]n2)C1 c1(C(=O)NCC2CC(NC(c3cc(Cl)no3)=O)CC2O)cccc(CO)n1 Cc1ccnc(CNC(=O)C(O)CNC(=O)C=Cc2ccco2)n1 C1(COC)CC(C(=O)NC(C)(C)CCNC(c2ccccc2C(C)C)=O)CCO1 c1(NC(=O)NCc2cccc(C#C)n2)ccc2c(c1)C(=O)N(C)CC2 N1(C(CCSC)=O)CCC(C2CN(C(C3CCC(C4CCCO4)O3)=O)C2)CC1 C#Cc1ccc(C(=O)NCC(F)CNC(=O)CCOCC(C)C)cc1 N1(C(CC2(C)CC2)=O)C2CC1CN(C(c1cncnc1C1CC1)=O)C2 c1(C(=O)NCCCCCOC2CCCCC2)ccc(Br)c([N+](=O)[O-])c1 C1(NC(C2N(C)CCC2)=O)CCC(C(=O)NCc2nccnc2Cl)CC1 CCCCCCC(=O)NCC(O)CN(C)C(c1cc(F)c[nH]1)=O CC1CN(C(=O)Cc2cccc(F)n2)CC(CCNC(C2(C)COCCO2)=O)O1 CCC(CN(C)C)CC(=O)N1CC(CNC(=O)CCN2CCC(N(C)C)CC2)C1 CN1N=CC(CC(N2CC(F)(CNC(=O)CCCc3cccc(Cl)c3)C2)=O)C1=O N1(C(=O)OC(C)(C)C)CCCC2(CCN(CCCN3CC4CCC3C4)C2)C1 C1(COCC)(CNC(=O)C(C)OC)CCN(C(=O)COC2CC(F)(F)C2)C1 C(=O)(CCC(C(=O)NOCc1ccc(C)cc1)NC(=O)CCOC1COC1)OC N1(c2cc(C(=O)OC)ncn2)CCCC2C(NC(=O)C(O)CSC)C(C)(C)C12 C1(C(N2CCC(c3nn[nH]n3)C2)=O)CCN(C(=O)CCCC2CC2)C12CC2 c1(C(=O)NCC(F)(F)F)ccsc1NC(C1CCC1CNC(C1C(=C)C1)=O)=O C12(CNC(=O)C(=O)Nc3cc(CN(C)CC)ccn3)CC3CC(C1)CC(Cl)(C3)C2 C1(C(=O)NCCOCCO)(COC)C=CCN1C(=O)C(C)Nc1ccccn1 C(CC(O)C(=O)NCCN(C(=O)C=Cc1ccc(SC)s1)C(C)C)SC C(=O)(C(C)CN(C(=O)CCc1nc(O)n[nH]1)C)NC(c1cccs1)C Cc1cc(C(c2nnnn2Cc2ccccc2)NC(C)C(=O)N(C)C)nc(C)n1 C1(NC(c2cc(CC)[nH]n2)=O)CC2CC(NC(c3cncc(NC)c3)=O)C2C1 N1(C(C(CC)=CC)=O)CCC2(CCN(C(=O)CN3CCn4ccnc4C3)C2)C1 c1(OC)ccc(C(=O)N(CCNC(C2CCC(C(=O)OC)CC2)=O)C2CC2)nn1 Cc1c(NC(=O)NC2CN(C(C3CCCCC3(F)F)=O)C2)cccc1Cl C1(C(=O)NCC(C)(F)CNC(=O)COCC(N2CCCC2)C)(OC)CCOC1 CCCC(CC1CCCC1)C(=O)NC1CCC1C1CCCO1 C=C1CCC1C(=O)NCC1(N(C(=O)C=CC2CC2)CC)CC1 c1(OC)ccc(F)c2cc(C(=O)NCCNC(=O)CC3(C)CCS(=O)(=O)N3)[nH]c12 c1(C(=O)NC2COCCN(Cc3cnc(CCC)s3)C2)cc(O)c(O)c(O)c1 c1(C(N(C2CN(C(COC(C)=O)=O)CC2O)C)=O)c(C)nc(C(C)C)nc1O Cc1ccc(NC(=O)CNC(=O)CNC(=O)C(c2scnc2C)N)c(Cl)c1 C#Cc1c[nH]nc1C(=O)NCC#CC(N1CC(C)CC1CC)=O C12(C(=O)NCCc3cnc(C)s3)CCC1CN(C(=O)CCc1ccn(C)c1)C2 N#CCCCC(=O)N1CC2C(NC(c3ccnc(C4CC4)n3)=O)C2C1 N1(CCC(=O)NCCCN(C(C(C(C)OC)O)=O)C)C(=O)NC2(CCCC2)C1=O c1(C(=O)NC(C)CCNC(c2cccc(CF)c2)=O)cc2c(F)ccc(Cl)c2[nH]1 CCCC(CCNC(C1CN(C(C2(C)CC3C=CC2C3)=O)CC1CC)=O)CCC c1(C(=O)NC2C(C(N(C3CCCC3O)CC)=O)CCC2)n[nH]c2ccccc12 c1(C(N(C)CCOCCNC(C2CC(F)C2)=O)=O)cnn(CC(F)(F)F)c1 C1(C(=O)NCC(C(C)O)C)CCN(C(=O)C(C)C#N)O1 N1(C(=O)NCC(CC(C)C(F)F)C)CCC2CCCC12CO.C(C)(C)(C)O c1(C(=O)NC2C(OC)CN(C(=O)CCC(=O)c3ccc[nH]3)C2)cc(C)nc(C)c1 C1(NC(C(CCC)=CCC)=O)CN(C(=O)C2=CC(C)(CC)C2)CC1C1CC1 C1(NC(C(COC)OC)=O)CCCC(C(=O)NCC=C(C)C)C1.C(C)(=O)O Cc1csc2ncnc(N3CCC(NC(C4CCCC5(CC5)C4)=O)C34CCC4)c12 c1(C(CCCNC(c2n(C)cc(Cl)c2)=O)=O)ccc2c(c1)CCCO2 Cc1cnc(CCCC(=O)NC(c2csc(C)n2)C)[nH]1 C1(NC(C2CCN(C)C2)=O)CN(C(C2(F)CCCCC2)=O)CC2(CCC2)C1 O=C(CCCCCNC(c1cnn2c1CCC2)=O)NCC(F)Br C1(S(C)(=O)=O)(C(=O)NCCOCCCNC(C=C(CC)CC)=O)CCC1 N1(C(C2CC(SC)C2)=O)CCC(CCCCNC(c2nc(C)c(C)s2)=O)CC1 C(C(=O)NC(C)(C)C(=O)NCC=C(Cl)Cl)(C(C)C)SC Cc1cccc2nc(C(N3CC(NC(C4(F)CC4C)=O)C(O)C3)=O)cn12 c1(C(N2CCOC(C(N3CCOC(c4nn[nH]n4)C3)=O)C2)=O)cccc(F)c1 C1(NC(C(=Cc2cccs2)C)=O)CC(NC(C2COC(C)C2)=O)CC1O c1(CC)ccc(C(=O)NC2(C3CCCN3C(c3cncn3C)=O)CC2)c(C)n1 N1(C(c2n(CC)ncc2)=O)CCC(CCCNc2ncncc2Br)CC1 c1(-c2ccc(C)nc2)cc(S(=O)(=O)N2CCN(C(C)C)CC2)c(C)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)C1)=O)NCCC(C(=O)OC)O c1(C(=O)NC2CCC(CNC(C3C(C)=C3)=O)C2)cccc2nc(C)sc12 C1(c2onc(CCNC(COCc3ccccc3)CO)n2)(CC)CCOCC1 S(=O)(=O)(c1ccccc1)NC(C(=O)N(CC(C)N)Cc1ccc(N(C)C)cc1)=O N#CC1(C(=O)NCC2CCN(C(c3cn(C4CCOCC4)nn3)=O)C2)CCCO1 S(=O)(=O)(c1ccc2c(c1)CCC2)N1CCC2(CN(C(C3C(C)C3)=O)C2)C1 N1(C(C=CCC)=O)CCC12CN(C(c1cn(-c3ncccn3)cn1)=O)C2 Cc1ncc(CCC(N2CCSCC2CCNC(c2conc2C)=O)=O)c(O)n1 c1(C(N2CCCC(CNC(C3CC(OC)C3)=O)CC2)=O)nn(C)c2c1CCC2 CCCC(C)(C)CC(=O)N(C1CCCN(C(c2sc(C)nc2C)=O)C1)CCO c1(OC)c(C(=O)NC(C)(C)CCNC(c2cnc(C(C)C)s2)=O)csc1Cl N1(C(C(CC)C(F)(F)F)=O)CCN2CCN(C(=O)CC3CCOC3)CC2C1 c1(C(=O)NC2CC(CNC(C(CC)(C)C(N)=O)=O)C2)ccc2cnn(C)c2c1 c1(C(=O)NC(C)CCNC(C2(n3cncn3)CC2)=O)cnc(Cl)cc1N C=CC1CN(C(c2ncccc2O)=O)CC1NC(C1CC2(CCCO2)C1)=O c1(C(N2C(C)CCC(NC(c3c(C)nn(C)c3C)=O)C2)=O)cc(Cl)c(F)cc1O N1(C(C(C)OC)=O)CC(CNC(c2ccc(Br)c(F)c2)=O)C(C)(C)C1 n1(CC(=C)C)nnnc1C(c1cc(C)ns1)NCc1nocc1C(C)C c1(C(=O)NC2CCC(N(C(=O)CSC3CC3)C)CC2)cccc2c1CCC2=O c1(C2(C(=O)NC3CCCC(CNC(C4(CO)CC4)=O)C3)CC2)c(Cl)cccc1Cl CCC(O)C(C)(C)C(=O)NC1C2CC(NC(=O)C(C)C(F)(F)F)CC12 N1(C(CCc2cc(OC)c(Cl)cc2)=O)CCOC2CN(C(C3CC3C)=O)CC12 Cc1ccc(C)c(CN2CCC(O)CC2C(N2CCC(CCO)CC2)=O)c1 O=C1OC2CC(C(=O)NC3CCCC(NC(=O)Cc4cnc[nH]4)C3)CC2O1 N1(Cc2cn(CC3CC(N)C3)nn2)CCC2(CC1)OCCc1ccccc12 N1(C(C(C(=O)OCC)CC)=O)CCCN(C(c2cn(C(C)(C)C)nn2)=O)CCC1 C=CCC(CNC(=O)C(C)NC(c1cccs1)=O)NC(c1ccco1)=O CCCC(CNC(C1(C#N)CCOCC1)=O)C(=O)NC1(CO)CC(OC)C1 N1(Cc2cn(CCCNC(COC3C(C)(C)CC3)=O)nn2)C(=O)CNC1=O N1(C(c2ccc(CNC(c3n[nH]c(C)c3C)=O)o2)=O)CC(F)(C2CC2)C1 c1(COC)nn(C)cc1C(=O)NCC1(F)CCN(C(C2CC(SC)C2)=O)C1 C(CC(C(C)C)NC(=O)Nc1ccccc1CNC(C1(N=[N+]=[N-])CC1)=O)OC c1(C(N2CC(NC(c3cccc(CC)n3)=O)C2)=O)cc(Br)c(O)nn1 C1(F)(CNC(c2ccc(C(F)F)o2)=O)CCCN(C(c2ccccn2)=O)C1 N1(C(C2CCC(C)NC2=O)=O)CC2CN(C(=O)C(F)CC3CCCC3)CC2C1 C(=O)(CCCC(=O)N1CCOCC(CNC(=O)CCC2CC2C)C1)N(CC)CC Cc1nc(N(S(=O)(=O)Cc2cnn(-c3ccccc3)c2)C)n[nH]1 CC1CN2CCN1CC2C(=O)NCCCN(C)C(c1ccoc1)=O C1(C(=O)NCC2N(C(CSC(C)C)=O)CCCCC2)CCn2ccnc2C1 c1(C(=O)NCCC(C)(CC)NC(C(CC)OC)=O)ccnc2ccncc12 c1(C(=O)NC(C2CCN(C(c3scc(C)c3)=O)C2)C)sc2nccnc2c1N C1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)n2cccn2)COCCC1(F)F N1(C(C(OCC)OCC)=O)CCC(OC(C)C(=O)NC2CC(Cl)(Cl)C2)C1 C1(C(=O)NC(c2ccc(Br)s2)C)C2CC(CC2F)N1C(C1CCC=CO1)=O C(CN=C(NCCN1CCOCC1)NCc1nnc(C)s1)c1c(C)cccc1.O N1(CC)CCC(NC(N2CCC(CC(C)CO)CC2)=O)CC1 c1(OC)cnccc1C(N1CC(CC(=O)NC2CC=C(C)CC2)CC1C)=O Cc1cc(C)c(C(=O)NC(C2CCCCC2)CNC(=O)CC2CC(C(F)F)C2)s1 N1(C(Cc2c(NC(c3c(C)n[nH]c3)=O)cccc2)=O)CCCCC(S(C)(=O)=O)C1 C(=O)(C(CC)CC)N1C(COCCCN(C(C(C)OCC#C)=O)C)CCC1 c1(CCC(N2CC(COC)C(N3CCOCC3)C2)=O)cccc(Br)c1Cl c1(C2N(C(c3cc(Br)c(Cl)s3)C(=O)NC3CCC3)CCC2)ccc(F)cc1 c1(C(=O)NC2C(C)CN(C(C3(CO)CCC3)=O)CC2)ccc(=O)n2c1CCCC2 N1(C(C2N(C(c3cc(CC)oc3C)=O)CC(=O)N2)=O)CCN(C2CC2)C(C)C1 c1(CNC(N(CCC)C2CC2)=O)ccc(Oc2cccc(C(F)(F)F)c2)nc1 C1(CC)COCC1N=c1nc2sccc2c(N(CC(C)N(C)C(C)=O)C)[nH]1 CC1CCCN(C(=O)Cc2ccn(C)n2)C1CCN=c1[nH]ncs1 C1(NC(C(C)=CC2CC2)=O)CC(NC(=O)Cc2sccc2C)CC1O C1(CNC(=O)C(F)Cl)CC12CCN(C(c1ccccc1-n1cncn1)=O)CC2 c1(C(=O)NC(C)CNC(c2ccccc2C(C)(C)C)=O)cn2c(n1)COCC2 N1(CC)CC(C(N2CCC(C)(CCNC(=O)CCOC)C2)=O)CCC1=O C1(CC=C)(NC(C2CC(C)C2)=O)CCN(C(C2COC3(CCC3)C2)=O)CC1 c1(CCC)noc2nc(C)cc(C(=O)NCC3CC(O)CN3C(=O)C3=CCC3)c12 c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)C2)C)c(C)nc(C)n1O c1(C(=O)NCC2C(NC(CC(C)C)=O)CCC2)ccc(OC(F)(F)F)cc1 CC(C)C#CC(=O)NCCSCCn1cc(COCCO)nn1 c1(C(N2CCN(C(C(CC=CCC)C)=O)C(CCO)C2)=O)cc([N+](=O)[O-])c(C)s1 C(CC(C)(C)CO)NC(C(C)CNC(c1ccc(Cl)s1)=O)=O C1(C(=O)NC(c2cccnc2)CC)CCN(C(=O)CN2CCCC2)C12CCC2 C(=O)(C(C)S(C)(=O)=O)N1CC(CC)C(C(=O)NCC(O)CC2CCC2)C1 c1(C(N(C(CNC(c2cn(CCC)nc2C)=O)C)CC)=O)cc(OC)ccc1C CC1CCC(N(C(=O)CC2(CNC(c3cccn3C)=O)CC2)C)C1 c1(CNC(C2(CNC(C(C)n3cncn3)=O)CC2)=O)nocc1Br.C(C)(C)(C)C(=O)O c1(C(=O)NCC2C(NC(COCC=C)=O)C2)cc2cnccc2cc1F c1(C(N(CC(C)N(C(C2(SC)CCC2)=O)C)C)=O)ccc(C(F)(F)F)cc1N c1(C(=O)NC2CCCN(CC(=O)NCCNC(N)=O)C2)cc(F)ccc1Cl c1ccc2c(c1)CC2CCNC1CCN(CC2CCOC2)CC1 c1(C(N2CC(NC(C3(CC)CC3)=O)C3C2C3)=O)c(C)nn(C)c1C CC#CCC(C(=O)NCc1cccc(Cl)c1)NC(=O)Cc1ccc(C)s1 CC1(C)CCN(CC(N2CCOC(c3cn(CCCSS(C)(=O)=O)nn3)C2)=O)C1 Cc1nn(CC(C(F)(F)F)NC(=O)C(=O)NC2CCOC2)c(C)c1C.C1CCO1 C(CCCCC(=O)NCCCN1CCCC1)n1cc(-c2c(CC)cccc2)nn1 Cc1cc2n(n1)CCN(C(=O)CC1COCCN1C(c1cc(O)no1)=O)C2 C1(C(N(C2CCN(C(=O)C=Cc3ccncn3)C2)C)=O)CCC2CCCCN12 C1(O)(C(C)NC(=O)CC(C)C2CCCO2)CCN(C(C2(O)CCSC2)=O)CC1 N1(C(c2cn(C)nc2CNC(=O)CC2C=CCCC2)=O)CCC(C)(CO)C1 C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NC(C)CCCNC(=O)CSCCC#N C1(C(N(CCC)CCNC(=O)CC2COC3CC2C3)=O)CSc2ccccc2O1 C(=O)(CCC(=O)NCC1COCCN1C(c1ccoc1Br)=O)NC C(C(=O)N=c1nc(C)[nH]n1-c1ccccn1)OCCC c1(CC(=O)NC(C2CCOC2)CNC(CC=C)=O)cnc(C)nc1O CC(O)CCCCCC(=O)NCC(O)CNC(=O)CCCC(N)=O c1(OC)ccc(C(C)(C)CNC(c2cn(C)nc2OC)=O)cc1F C1(C(CC)(C)C)CCC(C(c2nnnn2C(C)(C)C)(C)NCC2CC=CC2)CC1 CC1OCCCC1C(=O)Nc1ccc(-n2nc(C(C)(C)C)cc2C2CC2)nc1 CC(N=c1nc(C2CCCC2)[nH]s1)C1CCN(C(=O)CN(S(C)(=O)=O)C)C1 C(CC(O)C(=O)N(C1CC(C(=O)NCC(C)(O)CO)C1)C)N(C)C C1(NC(c2ccc(CNC(c3c(C)nsc3N)=O)cc2)=O)CC(=O)NC1(C)C c1(C(=O)NCCC(C)N(C(C(C2CCCC2)OC)=O)C)ccc([N+](=O)[O-])n1C Cc1cc(F)c2cc(C(N3CCC(C)(C)C3CNC(=O)C(C)CO)=O)[nH]c2c1 c1(C(=O)NCc2c(C(=O)NC(C)CC3CC3)occ2)ccc([N+](=O)[O-])o1 C(=O)(C(CC(C)C)C(C)C)NCC(CC(C)C)NC(c1cc2c(nn1)CCC2)=O c1(-n2c(Cc3n[nH]c(C)n3)nc(CCOC)n2)ccc(C)c(F)c1 c1(C(CN(C(=O)Cc2cnnn2C)CC)NC(CC=C=C)=O)ccc(C(C)C)cc1 Cc1cc(=O)c(C(=O)NC2CN(C(=O)C(C)n3cccn3)CCC2C)cn1C C1(C(NOCCC#C)=O)CCC(C)(C)N(C(C2CC(OCC)C2)=O)C1 CCCCC(C(=O)N1CCC(C)(C)C(C(=O)NCC(OC(C)=O)OC)C1)C(C)C Cc1ncc2ccccc2c1C(=O)NC(C1CN(CC2(CS(C)(=O)=O)CC2)C1)C CCCS(=O)(=O)C(C)C(=O)N1CC(C)(NC(=O)C=C2CCN(C)CC2)C1 C=CC(C(=O)NCC(C)(CO)NC(c1coc(N(C)C)n1)=O)OC CCC(F)(F)C(C)(C)C(=O)NCC(C)(C)CNC(c1cc(-c2ccco2)cs1)=O c12sc(=N)[nH]c1C(=O)NC(CO)C(C)NC2=O.c1(CC)nc(C)[nH]c1C(F)(F)F N1(C(C2=NOC(C)C2)=O)CCC(NC(=O)CCc2cncs2)C(F)(F)CC1 c1(C(=O)NCc2csc(-c3cc(Br)cs3)n2)ccc(OC2CC2)cc1 Cc1cc(CCC(=O)NC(CNC(=O)CCc2cc[nH]n2)CO)cc(C)n1 O=C1C2C(c3ccc4c(c3)CCCO4)CCN2C(=O)N1CCF C(=O)(C1CCc2nccn21)NCC1C(C(=O)NCC2(C)CC(C)(C)C2)CC1 N1(CC(=O)N(c2scnc2C)C(C=C)C)CC2(CN(CC(=O)OCC)CCO2)C1 C1(C(=O)NC(CC)CC)CC2CCN(C(=O)CCc3nc(C)cs3)CC12 C=CC(O)C(C)(C)C(=O)N1CC2C(C1)N2C(=O)Cc1cc(F)cc(F)c1F CC1CN(C(=O)CC2CCSCC2)CC1NC(C1OCCC1Cn1ccnc1)=O c1(OCC)cnc(C(=O)Nc2c(NC(C3(F)CCCCC3)=O)c[nH]n2)cn1 CCCCC(O)CC(=O)N(C)CC1(O)CCN(C(c2cc(Cl)n(C)n2)=O)C1 Cc1cnc(N2CCC=C(Cl)C2)c(S(=O)(=O)NC(C(C)C)c2ccco2)c1 Cc1csc(C=CC(N2CCC(CCNC(c3c(O)noc3C)=O)C2)=O)n1 C(=O)(C(F)CC(C)(C)NC(C1CC(F)(F)C1(C)C)=O)N(C)C C12CCN(CC1)C2.C(CCC(C)NC(=O)Cc1cn(Cc2n[nH]cc2C)nn1)SC C123C4C5C1C1C2C4C51C1(CC1)C(=O)NCC1CCCC(C1)NC3=O.COC N1(C(C=NOC)=O)CCCC2(CC(NC(c3ccc(OC)c(C)c3)=O)C2)C1 C(=O)(CCC1=CCCCC1)N1C(CCNC(C2(C(N(C)C)=O)CC2)=O)CCC1 N1(C(Cc2cn(C)nc2)=O)CC(NC(c2coc(CO)c2)=O)CC12CCCOC2 c1(C(=O)NC)ccnc2ncccc12.C12CCN(C1)C(=O)CNC2=O C=CCC(CC)C(=O)NCC(CC)N(C(=O)CC(O)Cc1ccccc1)C C1(O)(C(=O)NCCC(C(C)C)Nc2nccc(C)n2)CCCC(C)(C)CC1 c1(C(C(=O)O)N(C(C2C(C)C2)=O)C)ccccc1-c1ccccc1 c1(C(N2CCC(NC(Cc3nc(C)sc3C)=O)C(C)C2)=O)cc(N)c(O)c(F)c1 N1(C(CCC2CC(N(C(C(C)C)=O)CC(C)C)C2)=O)CCCCCC1CO C(CN=c1[nH]c(=NCc2nccnc2C)[nH]c2ccsc12)N(CC)CC C1(CF)CC(N=c2nc(NC3COc4cc(F)ccc43)c3c([nH]2)CSC3)C1 C1(C(=O)NC(CNC(CN(C(C)=O)C)=O)C)(C(F)F)CCCO1 CCC(C)C(C)C(=O)NCCCN(C(=O)Cc1cncc(C#N)c1)C C(=O)(CCCCC(N)=O)NC(C(=O)Nc1ccc(C)c(C)c1)(C)CO c1(-c2ccc(CC)cc2)ccc(S(=O)(=O)NC(C)CSC)cc1C C(=O)(C(C)(O)C(C)C)NCC12CC(NC(c3c(C)ncs3)=O)(C1)C2 C1(NC(C2CC(=O)N(O)C2)=O)C2CCC1N(C(c1ccc(F)o1)=O)C2 N1(C(C2C(c3c(C)ccs3)C2)=O)CCC(NC(C2CCCN2C)=O)C1 C(=O)(CC1OB(O)c2ccccc21)NCc1noc2c1CC(C(C)=O)CC2 C(C)(N=c1[nH]c(N2CCC3(CCC3)C2)nc2ncn(C)c12)c1c(C)cccc1F c1(C(N2CC(C#C)N(C(c3cc(CO)[nH]n3)=O)CC2)=O)cn(C)c2ccccc12 Cn1ncc(C#N)c1C(=O)N(C1CC1)CC1CCCN1C(=O)CCC1CCOC1 C1(OCC)CCCCC1C(=O)N(c1ccc(C)cc1)CCNc1ncc(C)cn1 c1(OC)ccc(O)c(COC(C2(C)CCCCN2C(=O)OC(C)(C)C)=O)c1 CC1(C)Cc2cccc(C(N3CCCCC(NC(C4CC4(C)Br)=O)C3)=O)c2O1 C#Cc1cccc(C(=O)N(C2CN(C(=O)CCC=CC(C)C)CC2O)C)c1Cl N1(C(c2c(C(N)=O)coc2)=O)CC(NC(=O)CC(=O)NC2CC2)C2(CC2)C1 Cc1cc(OCc2cn(CC3CCCN3C(=O)CC34COC(C3)C4)nn2)ccn1 C(=O)(C(CCC)C(C)C)NC(C(=O)NCc1nc(CC)[nH]n1)C(C)(C)O CCC(C)(F)C(=O)NCC(c1cccc(Br)c1)NC(C12CCC1CC2)=O C1(C(C2(CC)CC2)=O)CC2CC(=O)C1O2.C12CCC(C1)CNC2=O.NCC N1(C(CSCCOC)=O)CCCC(CO)(NC(C2CC(=O)N(C)C2)=O)C1 C1(CC(=O)NC(CNC(CCC=C)=O)C)CCN(C(=O)CN2CCSCC2)CC1 C1(C(=O)NC2CN(C(c3ccc(C)cc3N)=O)CC2O)Cc2cc(Cl)ccc2O1 S(=O)(=O)(c1cccc(Cl)c1F)N1C(C)(C(=O)Nc2ccc(C(C)=O)c(Cl)c2)CC1 N12CCN(CC1)n1cc(nn1)-c1ccc(o1)C2=O.C1CCN(C(=O)C(F)F)C1.CO c1(NCCCCCCCCC)cc(=NCC(C)CNC(=O)CCCCC)[nH]cn1 c1(C(N2CC(C)C(NC(c3noc4ncccc34)=O)C2)=O)cnc([N+](=O)[O-])n1C S(=O)(=O)(c1cccc(SC)c1)NCC(C)(O)C1(C(c2ccccc2)O)CC1.CO C(=O)(CC(C)(C)C(=O)N1CCCC2(NC(c3cc(C)no3)=O)CC2C1)OC c1(C(=O)NCCN(C(CC(C=C)C)=O)CC(C)O)cc(S(N)(=O)=O)cc(Cl)c1F Cc1noc(C)c1CC(=O)N(CCCNC(=O)COC1CCCCC1C)C O=C(CCC(CF)CF)NCCNC(C1CC2(C1)CC21CCC1)=O O(n1nnc2c1CCN(C(=O)OC(C)(C)C)C2)NC(c1cccc(=O)o1)=O N1(C(C2C(=C)C2)=O)CCN(C(c2ccc(C(F)F)nc2)=O)CC1C1CC1 c1(NC(C(C)CNC(c2nc[nH]n2)=O)=O)ccc[n+]([O-])c1 N1(C(C(c2scc(CC)n2)(F)F)=O)CCOC2(C1)CN(C(=O)C(F)(F)CO)C2 c1(NC(c2n(CC(=C)C)nnn2)(C)C(C)SC)cccc(-c2cncnc2)c1 C(=O)(C(C)CCCC(C)C)NC(CC=C)C.C12(CCCCC1)C(=O)N2 N1(C(c2scc(COC)c2)=O)CCN(C(=O)CC2(OC)CCC2)CC1C(C)(C)C C(=O)(CCCCCNC(N)=O)NCC1N(C(C=C(CC)CC)=O)CCC1C c1(C(=O)OC)ccc(O)c(CN2CC(OC)CC(C)C2)c1.N12CCCC1C2=O C1(CC(=O)NC2(CF)CCN(C(=O)CCn3ccccc3=O)C2)CCCCC1O c1(CCC)nc(=NC(CNC(C2CCSC2)=O)C2CC2)s[nH]1 O=C(C(O)CC(F)(F)F)N1C2CC1CN(C(c1cn(C3CC3)nn1)=O)C2 C1(COC)CN(C(=O)C(Cc2ccco2)NC(=O)C(C)Cn2cccn2)C1(C)C C1(C(=O)NC2CCN(C(c3ccns3)=O)C23CC3)CC12CCC(F)(F)CC2 c1(C(=O)Nc2cccc(CNC(CC3(COC)CC3)=O)c2)ccc(S(N)(=O)=O)o1 CC1(C)CC(C(=O)Nc2cncc(O)c2)CCN1C(C1CCC(C)(C)C1)=O C1(CC(=O)NCC(COC)NC(c2nc(Cl)oc2C)=O)C(=O)NN=C1C Cc1cc(=O)c(C(=O)NCC2CN(C)CCN2C(c2cc(O)cs2)=O)cn1C CC1(C)C(C(=O)N(CC(O)CF)CCO)C1CNC(=O)C(O)CC1C=NC=N1 C1(NC(C(C)NC(N)=O)=O)CCCCN(C(c2nc[nH]c2C(F)(F)F)=O)C1 c1(OC)cc(CNC(=O)C(C)C(=O)C(=O)SCC(C)N)cc(F)c1.C(C)(C)(C)O N1(C(c2cn(CC=C)nn2)=O)CCC(CC)C1CNC(=O)CC1CC1 C(c1ccc(C)cn1)=CC(=O)N(CCNC(=O)CCc1nccs1)CC c1(OCC(=O)N(CC(C)(C)NC(=O)CC2(C)CCOC2)C)ccc(F)cn1 c1(C(=O)NCC(C2CC2)NC(=O)C=CC=C(Cl)Cl)cnc(O)o1 c1(C(=O)NCCCCN(C)Cc2ccccc2-n2ccnn2)ccc([N+](=O)[O-])cc1 N1(C(C(CCC)NC(=O)CCCN(C)C(C)C)=O)CCNC(=O)C1CCO C(CC(C(C)C)NC(=O)CC1CCC(=O)N1)N(C(C=C(C)C)=O)C c1(C(=O)NCCC2CN(C(=O)C(O)C3CCC3)C2)ccc(Cl)c2occc12 c1(CNC(C2C3CN(C(C4(SC)CCC4)=O)C2C3)=O)sc2ccccc2c1C c1(C(N2C(C)CC(NC(c3nonc3N)=O)CC2)=O)cc2ccccc2cc1F CCC(C(=O)NC1CC(CNC(=O)C(C)(C)Oc2ccccc2)C1)C(C)O CC1(C)CCCC(CC(=O)NC2CCCC2CNC(c2csc(C3CC3)n2)=O)C1 C12(NC(c3cccc(N)c3)=O)CCCC1CN(C(c1coc(O)n1)=O)C2 C1(C(=O)NC2(C(N(CCCCOC)C)=O)CCCC2)CCC(F)CC1 C1(CC(=O)NC2CC2(F)F)COCCN1C(c1ccc(Oc2ccccc2)cn1)=O C#CCCN=C(NCC1CCCN1c1ccsc1)NC1CCOc2ccccc21 c1(CC)c(Cl)nc(C)[nH]c1=NCC=CCNC(C1CCC2CCCCN12)=O C1(CC=C)(NC(c2ccsc2C(F)F)=O)CCN(C(=O)COCCOC)CC1 N1(C(c2ccc(C(C)=O)o2)=O)CCC(C)(C)C1C(N1CC(OCC(C)C)C1)=O C1(C)(C(=O)OC)CCN(C(=NCCCCl)NCC(c2ccc(Cl)cc2)O)C1 C1(NC(c2nn(CC)nc2C)=O)CN(C(=O)C(F)C2CCCC2)CC1S(C)(=O)=O c1(CCC)cc(C(N2CC(NC(=O)C(C)=C3CC3)C2)=O)cc(O)n1 C1(NC(=O)OC(C)(C)C)CCCC1C(=O)COC(=O)CCCc1ccccn1 N1(C(CSCCN(CC=C)CC)=O)CC(O)(CNC(C2(C3CC=CCC3)CC2)=O)C1 C1(NC(c2nc(SC)sc2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC1C C1(C(=O)NC(CC=C)CNC(=O)C=C(C)C(C)C)CCC(=O)N1C(C)C n1(CC(N2CC(OC)C(NC(=O)Cc3ccns3)C2)=O)ccc2c(C)cccc12 C1(NC(CC2C(NC(C(CC)OC)=O)CCC2)=O)CCC(N(C)C)CC1 c1(NC(CC)(C)C)ccc(S(=O)(=O)NCCCN2CCCC2=O)c(Br)c1 C=CCC(C)(C)CCn1cc(CC(=O)NC(=O)C(Cc2ccsc2)NC=O)nn1 N1(C(CN(C(CCc2onc(C)n2)=O)CCO)=O)CCc2ccccc21 N1(C(c2c(C)n[nH]c2C)=O)C2CCC(C2)C1C(N1CC(CC2CC2)C1)=O C1(C)(CC(C(C)C)N(C)C)C(O)CN1C(=O)CCc1nccc(=N)[nH]1 C1(NC(c2ccoc2)=O)CCCC1NC(C1(c2ccccc2)CC(O)C1)=O CCCC(C(=O)N(C1CC(NC(=O)Cc2cccnc2Cl)C1)C)N(C)C c12ncnc(c1C)NCCC1CCN2C1.c1(CC2(COC)CC2)ccccc1 N1(C(CC(C(C)C)C)=O)CC2=C(C1)CN(C(C1CN(CP(C)(C)=O)C1)=O)C2 N1(C(C2=CC(O)C(C(C)(C)C)C2)=O)CCc2cc(Br)c(Br)cc2C1 N1(C(c2nc(N(C)C)oc2)=O)CCN(C(C2CCCNC2=O)=O)C(CO)C1 CCC(C)C(C)(O)CNC(C1CN(C(=O)CCC2OCCO2)CC1(C)C)=O C1(OC)CN(C(c2cc(C)sn2)=O)CC1NC(=O)Cc1ccon1 C1(CNC(C(n2cc(-c3ccc(N(C)C)cc3)nn2)C)=O)CCC(C)(C)C1 n1(CCC)nccc1C(=O)NCCc1ocnc1CNC(C1CNC(=O)O1)=O C1(CNC(=O)NCCc2ccc(O)cc2)(CF)CC12CCOCC2 c1(C(=O)NCC2CC3CN(C(CC=CC=C)=O)CC32)c(Cl)nc2sc(C)cn12 C1(NC(CC2C(C)C2)=O)CC2CN(C(=O)CCC(=O)N(C)C)CC12 C1(CC)(NC(c2ccc(OC)nn2)=O)CCCN(C(C2CCCC23CCC3)=O)C1 C(=O)(CCC(F)(F)C(F)F)NC1(C)CC(NC(=O)C(C)(C)n2cnnn2)C1 C1(C(=O)NCC(C)(C)CNC(=O)Cc2cncnc2O)CC2(C1)CC1(CCC1)C2 C1(CNC(c2sccc2Br)=O)CN(C(=O)CCN2CCCC2=O)CCO1 Cc1cc(C(N2CC3CC2C3CNC(=O)Cc2ncoc2C)=O)c(Br)s1 C1(C(=O)NC(c2ncc(C)[nH]2)C)CCCN(C(=O)C(C)(C)C2CCC2)CC1 N1(C(C(C)(C)N2CCOCC2)=O)CCC2C1CCCN2C(C1C2CCCCC12)=O C1(CNC(c2cc(C)c(C)s2)=O)CCCN(C(c2cc[nH]c2)=O)CC1 C=CCC(C)C(=O)N1CCC(N2CCC(NC(c3snnc3CC)=O)C2)CC1 CCC(C)CCC(=O)NCC(C)(C)NC(c1csc(=N)[nH]1)=O C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CCCN(C(C(CC)OC)=O)C(CO)C1 C(=O)(C1c2ccccc2C(=O)N1C)N(CCCNC(=O)C(C)(C)c1cnc[nH]1)C c1(CC(=O)NC2(Cc3ccccc3)CC2)nccnc1O.C12CC(C1)CNC2=O CC(C)(C(=O)N1CCCC(C(C)(O)CNC(=O)Cn2ncnn2)C1)S(C)(=O)=O C(=O)(C(N=[N+]=[N-])C(C)C)NC(COCC)C(=O)NC1CC2OC1C1CC21 c1(NC(C(=O)N(C)CCN2CCCCC2O)=O)ccc(Cl)c(Br)c1F CC(C)CC(C)CC(=O)N1CC(NC(c2occc2Br)=O)CC1C C1(NC(=O)CCn2ccnn2)CCOC(C(=O)NCCn2cnnc2)C1 N1(C(C2CN(CC)C(=O)C2)=O)CC(NC(=O)COCC(F)F)C(C2CC2)C1 c1(C(C)C)nc(N2CC(N(C(=O)CN3CCC3)C)C2)c2cc[nH]c2n1 C1(c2cn(-c3ncc(Br)s3)nn2)(N(C)C)CCN(C(=O)CCc2ccccn2)C1 c1(OC)cc(CNC(c2cccnc2O)c2nnnn2C2(C)CC2)ccc1Br c1(C(N2CC(NC(C(C=C)CC)=O)C(SC)C2)=O)nc(C)ncc1Cl C(C1CCCCCC1)=CC(=O)NCC(CNC(C(c1c(C)noc1C)C)=O)F N1(c2[nH]c(=NCc3nn(C)c(Cl)c3)[nH]c(=N)n2)CCc2[nH]c(=N)nc(O)c2C1 C1(C(=O)NC2CC(CNC(COC)=O)C2)CCCC(Cc2ccccc2)C1 Cc1ccc(C(N2CCCCC(NC(c3cc(N)ccc3O)=O)C2)=O)cc1C c1(COC)sccc1C(=O)NC(C)CNC(=O)CC1(C)CC1(Cl)Cl CC1=C(C(=O)NC2CN(C(c3ccc(C(N)=O)[nH]3)=O)CC2(C)C)CCC1 c1(C(=O)NCC2C(C)CN(C(=O)CCCF)C2)ccnc2[nH]cnc12 N1(C(CC2N(CC)CCC2)=O)CCOCC1C(=O)NCC(=O)NC(C)C c1(OCCOC)cn(C)nc1OCCCOCC(=O)NCc1ccccc1 c1(C(N(C2CCN(CC)C2)c2nnnn2C2CC2)=O)cn2ccsc2n1 Cc1c(C(N2CC3CN(C(C4CCNC(=O)C4)=O)C3C2)=O)cc(F)cc1Br c1(C(N2CCC(NC(c3ccc(O)c(F)c3)=O)(CF)C2)=O)cnc2[nH]cncc1-2 Cc1cc(NC(C2CCC=CC2NC(=O)C2=CCSC2)=O)ccc1F C1(NC(CC2(C=C)CC2)=O)CCCC(NC(=O)Cc2cccc(C)c2)C1 c1(C(=O)NCCN(C(C=C(CCC)C)=O)CC)c(OCC)cccc1C N1(CCCNC(CC2CC(=C)C2)=O)CCC(NC(=O)CNC(c2occc2C)=O)C1 CC(C)CC(O)CC(=O)N(CC(C)C(=O)NCCCNC(N)=O)C c1(NC(C2CCCC(NCc3c(Cl)ccc(C)c3)C2)=O)c(Cl)cc(Br)c(Cl)c1Br Cc1c(C(=O)NCC2CN(C(=O)C3=CC(C)CC3)C2)[nH]c2ccccc12 c1(C(=O)NC2CN(C(CC(C)(C)OC)=O)C(C)C2)c(N)c(F)cc(F)c1F CC1(C)CC=C(C(=O)NCc2csc(C(=O)NC3CC3c3ccsc3)c2)CC1 C1(C(N(CCN(C(CN(C(=O)OCC)C)=O)C2CC2)C)=O)CCC(CC)CC1 c1(CCC(=O)NC2(C)CCN(C(C3CC3c3ccco3)=O)C2)ccc(C#N)cc1 N1(C(C2CCN(OC)CC2)=O)CCCC1C1CCCCN1C(=O)CC(C)C c1(CC(N2C(CNC(C3C4COCC34)=O)COCC2)=O)ccc(Cl)cc1F C(CC(C)C(=O)N1CCC(C(=O)NC2(CO)CCC2)C1)=CC CC(C)CC(C(=O)N1CCN(C(=O)CCC(C)N(C)C)CC1CCO)N(C)C C(=O)(C(C)(C)C(C)(F)F)N(CCNC(c1snc(-c2ccccc2)c1N)=O)CC Cc1c(C(N2CC(CNC(C3(C)CCCO3)=O)C(C)C2)=O)sc2cncn12 c1(CC(C(=O)N(CCC)CCNC(C2(NC(N)=O)CC2)=O)O)cccc(Cl)c1 C1(C(N(C2CCCCC2)CCNC(C(CC)C)=O)=O)COc2cc(F)ccc2O1 N1(C(CC(CC)SC)=O)CC(NC(c2cnc(O)cc2C)=O)CC1(CC)CC C(CC(C(C)C)NC(C1(CF)CC(F)(F)C1)=O)NC(C(C=CCCC)O)=O C1(CNC(CC=CCC)=O)C(C)CCN1C(=O)CCCNC(N)=O Cc1[nH]c2cccnc2c1C(=O)NCc1ncnc(Cl)c1CN1CCOCC1 C1(NC(C2(OC)CCC2)=O)CCCCCN(C(=O)Cc2cnns2)C1 N1(C(=O)C(O)CCCNC(=O)C(F)(F)CO)CCCC2(CCCO2)C1 C(=O)(CC(C(C)C)C(C)C)NCC1(C)C(C)CN(C(C(C(C)C)NC(C)=O)=O)C1 CCCCCC(CC)C(=O)NCC1CN(CCC2=CCCCC2)CCC1(F)F C1(O)(CCNC(CCCOC)=O)CCCN(C(c2sccc2OC)=O)C1 N12CCCC3CN(CC13)c1nc(ns1)C2=O.c1(CCOC)cc(C(=O)OC)no1 C1(C(=O)NC(C2CN(C(c3cc(-c4ccco4)[nH]n3)=O)C2)C)OCCN(C)C1=O c1(CC)cc(C)c(C(=O)NCCNC(C2(c3ccccc3F)CCC2)=O)o1 Cc1cc2cccc(C(=O)NC3(C(=O)Nc4cccc(F)n4)CC3)c2[nH]1 N1(C(Cn2c(C)ncc2)=O)CC(C)(C)CC1C(=O)NC1CC1c1ccsc1 N1(C(Cc2c(C)con2)=O)CCCCC1C1CCN(C(=O)C(O)C2CCCC2)C1 N1(C(CN(C2CCC2)C)=O)CC2(CCCC2NC(C2CCC(N(C)C)CC2)=O)C1 C1(N(C(=O)C=Cc2cn[nH]c2)CC)CCC(NC(=O)C(F)OC(F)(F)F)CC1 Cc1nc(C)c(C(=O)NC2(CF)CCN(C(=O)C(O)CC3CC3)C2)o1 c1(C(N2CCC(C)(CNC(C3CC=CCC3)=O)C2)=O)cc(F)cc(F)c1O N1(C(COCC#C)=O)CC(NC(=O)Cc2ccc(F)cn2)C(C)C1 N1(C(CCc2n(C)ncc2)=O)CCC(C(N2CCC2)=O)(CF)C1 C1(C2CN(C(=O)CC3CCNC(=O)C3)C2)(NC(C(c2c(C)n[nH]c2C)C)=O)CC1 CCC(CC(=O)NC1CN(C(=O)Cc2ccoc2C)CC1OC)SC Cc1cn(CC(=O)NC(C)(C)C(C)NC(=O)C=CS(C)=O)nc1C(F)(F)F C(=O)(CS(N)(=O)=O)NCC1(COC)CCCN1C(=O)C=C(C)c1cccs1 N1(C(C(=O)NCCCc2nccc(C)c2)=O)CCC12CCCC(C)(C)C2 c1(C(=O)NCCOCC(=O)N(CCCC)CCO)oncc1C N1(C(C(C)OCCOCC)=O)CCCN(C(c2nc(Cl)cs2)=O)CC1C(C)C S(=O)(=O)(CC(=O)N(c1ccccc1F)C)NC.C12CCC(N1)NC2 c12ccc3nc(sc3c1)N1CCC(CC1)C(C)O2.c1(C(=O)NCC)cscn1 CC#CCCCC(=O)NC(COCC)C(=O)NCC1(CC)CCOC1 c12cnc(O)c(c1)C(=O)N2.C1(C)(NC(C2CN(C(C)=O)C2)=O)CC1(F)Cl C1(C(=O)NC2CN(C(C(CC=C)C)=O)CC3(C2)CC3)CCc2nnc(O)n2C1 CC(C)C#CC(=O)N1CC(O)CC1CNC(c1cc(Cl)ccn1)=O CCC(C)CCCC(=O)NCC(=O)NCC(=O)N(C)Cc1csc(C)n1 c1(N(CCN(C(C(CC)OCC)=O)C)C(C)C)cc(C)ncc1C#N N1(c2n(CCC=C)c(Cc3cccs3)nn2)CCC2(CCC(=O)N2)C1 N1(C(c2c(NC(Cc3nc(C)[nH]n3)=O)cn(C)n2)=O)CCCC(O)(C(F)(F)F)C1 c1(C(=O)NCC2CC(NC(C3(CCC)CC3)=O)C2)cnn2c1OCC(O)C2 Cc1ncc(Cl)cc1NC(C1CC(O)CN1C(c1cnon1)=O)=O c1(NC(C)=O)ccc(C(=O)NC2CC(NC(C3(CF)CCC3)=O)C(O)C2)nc1 C=CCC(C)(O)C(=O)N1CCCC(N(C)C(c2ccc(OC)cc2F)=O)C1 c1(OC)ccc(-n2nc(CS(C)(=O)=O)nc2C(C(=O)OC)OC(C)C)cc1 C1(CC)COC(C)(C)CN1C(C12CC(CN(C(c3ncncc3C)=O)C1)C2)=O CC1(C)CC(CC(=O)NCCN2CCOCC2)N(C(C2(C)C(C)(C)C2(C)C)=O)C1 C(=O)(C(C)CC(=O)NC1CCCC(C(=O)NC2(C)CCC(C)(C)C2)C1)OC C(=O)(C1=CC2C=CC1C2)N(C1CCCN(C(Cc2ccn(C)n2)=O)C1)CCO N1(C(C(CC)C)C(=O)NC2CC(F)(F)C2)CCC=C(c2ccccc2O)C1 c1(C(=O)NCC(C)NC(C(c2ccccc2)NC(C)=O)=O)cc2c(ccn2C)s1 Cc1cc(-n2cc(CC(C)(N)C(N3CC(O)CC3(C)C(=O)O)=O)nn2)cc(C)c1 c1(C(=O)Nc2cc(OC)c(CN(C)C)cc2)ccc2ncnn2c1 c1(C(=O)NC2C(CC)CN(C(=O)Cc3cnnn3C)CC2)cc(C)c(F)c(C)c1 N1(C(C(C)CN2CCOCC2)=O)CCCC(C)C1CNC(C1COC(=O)O1)=O c1(C(=O)NCC2CC(NC(CSCC)=O)C2)cn(C)nc1C c1(COC)nnc2n1CCN(C(=O)CCC(O)C(F)(F)F)C2.c12cn(nn1)C(C)C2 N1(C(CC2C(C)C2)=O)C2CCC1CN(C(=O)CCc1nnc(S)n1C)C2 N1(c2nc(C)nc(O)c2)CC(NC(C2C3CC4C(C3)C24)=O)CC(C)(C)C1 N1(C(CCCSC)=O)CC2CCN(C(c3cccc(-c4ccncc4)c3)=O)C2C1 c1(CNC(CNC(=O)NC)=O)ncoc1C1CN(C(=O)Cc2cscn2)C1 CC1CCCn2ncc(C(=O)NCCC(C)CCNC(=O)CC3CC3)c21 N1(C(CCC(=O)NCC)=O)CCCC(F)(CNC(=O)C(=Cc2cnc[nH]2)C)C1 C12(CNC(c3c(C(C)C)ccs3)=O)CN(C(C3(C#N)CCC3)=O)CC1CCO2 CCCCC(F)C(=O)NCC(C)C(=O)NCc1nccc(C)n1 c1(CC(=O)N(C(CNC(CCc2cc(C)no2)=O)=O)C(C)C)ccc(C)c(Cl)c1 c1(NC(=O)Nc2cccc(NC(C)=O)c2)cccc2sc(Cl)nc12 C(=O)(C1=Cc2cc(C)ccc2OC1)NC1CN(C(c2n(CC)cnn2)=O)C2C1C2 C#CC1COCCN1C(c1ccc(F)cc1Br)C(=O)Nc1ccccc1C N1(C(CC(=C)C)=O)CCC(C(CO)NC(c2cc(OC)n[nH]2)=O)CC1 C1(CC(=O)N(C(CC(CC)C)C)C)CC2(C1)CN(C(c1ccn(C(F)F)n1)=O)C2 N1(C(CNC(=O)OCC=C)=O)CC(=O)NCC1C(=O)NCC1CN2CCC1C2 c1(COC)ccccc1CSc1cccc(NC(=O)NC2CC2)c1 C1(NC(C(C(C)OC)O)=O)(CO)CCN(C(=O)CC(=O)NCC2CC2)CC1 Cc1c(O)cc(C(N2CC3C(NC(=O)CC4CCC(=O)N4)C3C2)=O)cc1O C(C(C)C(=O)O)(c1ccccc1)NC(c1ccccc1F)C C#Cc1nc(C(=O)NCCC(C)N(C)C(C2CCOC2=O)=O)cs1 C(CCC(N)=O)(C(=O)N1CC2CC1CN2C(C1CC1F)=O)NC(C)=O CC(C)CC(F)C(=O)NC1CN(C(c2ccc(O)c(C(C)(C)C)c2)=O)C(C)(C)C1 C1(C(=O)NCCC(C)N(C(=O)CC(C)(F)F)C)CN(C(N)=O)CCO1 CC1CC(CNC(=O)Cc2cc(Cl)n(C)n2)CCN1C(=O)C(C1CCOCC1)O C1(NC(CCN(CCCCC)C)=O)C=CC(CNC(=O)C(=O)NC2CC2)C1 Cc1cccnc1C(C)NC(c1nc(CNC(C23CCC(C2)C3)=O)oc1C)=O C(=O)(C1CCc2nccn21)N1CC2(CCC(CNC(C(N)=O)=O)O2)C1 CCC(CC)C(C)C(=O)N1CCN(C(=O)CN(C)C(N)=O)C(C(C)C)C1 C1(OCC)CC2CN(C(C3C(C)CN3C(c3cn(C)cn3)=O)=O)CC12 C(=O)(C(C)(C1CC1)N(C(=O)CSc1ccccc1)C)NCCC(C)SC n1(CC)nc(C(=O)NCC2CN(C(C3CC(O)CN3C(C)=O)=O)CCO2)cc1O n1(CCCC)cc(C(=O)NCC(C)NC(c2cscc2CC)=O)nn1 Cc1nc(C)c(C(=O)NC(C)CN2CCN(C(=O)CC3CC(F)C3)CC2)c(C)n1 C(=O)(C1CCCc2ccnn21)N1CC2C(CNC(C3(CO)CC(C)(C)C3)=O)C2C1 C1(C#N)(C(=O)NC(CN(C(C(CCC)OC)=O)C)C)CCSCC1 n1(CCC)cc(CNC(=O)CCN(CCO)C(C2CC(=O)C2)=O)nn1 c1(C(=O)NC2CN(C(CC(=C)C)=O)C(C)CC2)cnc2n(c1=O)CCS2 c1(C(=O)OC)ccc(C(=O)NC(CO)C(C)NC(c2ccsc2C)=O)o1 C(=O)(C(=O)C(C)(C)C)N(C(c1cn(Cc2ccc(C(=O)O)o2)nn1)(C)C)C(C)C CCC(C)CCCC(=O)NCCCC1(NC(=O)C#CC2CCC2)CC1 C1(C)(CNC(C2(CCCC)CC2)=O)CCCN(C(c2ccc(O)cn2)=O)C1 C1(NC(C(C(C(C)C)O)C)=O)CC2CCCC(C1)N2C(c1ccc(F)cc1)=O c1(C(=O)NCC2C3CN(C(c4c(CC)noc4C)=O)CC32)ccc(C)c(F)c1N C1(C)(C(=O)NC2(C#C)CC3CCCC23)CCCN(CS(=O)(=O)CN(C)C)C1 c1(NC(C2CCC(C(=O)OC)CC2)=O)c(NC(N)=O)c(C(F)(F)F)nn1C c1(-c2c(F)c(C)c(F)c(F)c2)ccc2c(Cl)c(NC(=O)CC(C)O)cnc2c1 C1(C(=O)NCC(COC)OC)(COC)C=CCN1C(c1c[nH][nH]c1=N)=O C1(C(N2C(COC)CC2)=O)C(C)CCN1C(=O)CCCc1cnn[nH]1 N1(C(CC(C=C)C)=O)CCC2CN(c3ncnc(C(=O)OC)n3)CC2C1 Cc1noc(C)c1S(=O)(=O)Nc1ccc(C(=O)NCC2CCCC2N)cc1 c1(NC(N2CCCCCC2)=O)ccc(C(F)F)cn1.C12OCCC1C2 CC1CC(C(N)=O)N(C(C2CCC(c3cn(C4COCC4O)nn3)C2)=O)C1 Cc1cc2c(CC(N3CC(NC(C4CC(C)(C)CO4)=O)C(F)C3)=O)csc2s1 c1(-c2n(-c3nc(C)nn3C)nc(C3CC3)n2)ccc2ncn(C)c2c1.C(C)(C)CO N1(Cc2n(CC#C)ccc2)CCC(NC(=O)C(C)OCC(C)C)C(O)C1 N1(CC(=O)NCC2CC3(CC3)CN2C(C2CC2CF)=O)CCc2ccccc2C1 N1(C(C=CC(=O)N(CC=C)C)=O)CCCC1(C)C N1(C(C(C)N(C(=O)CC(C)(C)SC)CC)=O)CCC(C)(C2CC2)C1 C1(CCC(=O)OC)CCN(C(c2cnn(C)c2)C(=O)NCC2CC2)C1 c1(CC)cnc(Cl)nc1N1CCC(F)(CNC(=O)Cc2c(C)cccc2C)CC1 N1(C(C2(C)CC3CC3C2)=O)CCn2ncc(CNC(=O)C=CCO)c2C1 c1(C(C(=O)OCC)NC(C23CC(Cc4cccc(N)c4)(C2)C3)=O)ccc(F)cc1F C1(N(CC(=O)NCC2CC3CC3C2)C)CC(=O)N(c2nccs2)C1 Cc1cc(N)n2ncc(C(=O)NCCC(C)NC(C3CC4CCC(C3)O4)=O)c2n1 N1(C(CC2CC(OCC)C2)=O)CCC(C)(CNC(C2(C)CC2(F)Cl)=O)CC1 Cc1nc(C(=O)NCCC(C)N(C)C(C2CCOC2(C)C)=O)sc1C c1(SC)nn(C)cc1C(=O)NC1(C)CC(NC(=O)Cc2ncc(C)s2)C1 C1(C(=O)NC2CCC(NC(C34CC(C(C)C)(C3)C4)=O)C2)CC2CCC(C1)O2 CN(C)S(=O)(=O)NCC(=O)NCC1CC(O)CN1C(=O)CC(=O)NC1CC1 N1(C(Cc2cccc(SC)c2)=O)CC2COC(C)(C)OCC2C1 S(=O)(=O)(c1ccc(NCCc2ccccn2)c(C#N)c1)N(CC(O)C1CC1)C c1(C(N2CC(C)(NC(=O)C=Cc3nc[nH]n3)C2)=O)cc(C#N)c(F)cc1F CCCC(C#N)C(=O)NC1CC(C(F)F)(NC(=O)CC2(NC(C)=O)CC2)C1 C12(C(N(CCCNC(c3c(OC)cc(O)nc3)=O)C)=O)OCCCC1C2(F)F c1(OC)cccc(Cl)c1C(=O)NCCC1CC(NC(c2ccc(O)cc2F)=O)C1 N1(C(=O)NCC(CC(C)C)(C)N(C)C)CC23CCCC2(COC3)C1 C1(NC(=O)C=C(C2CC2)C2CC2)CC1C1CCCN(C(=O)Cc2nncs2)C1 C1(NC(c2c[nH]nc2C(F)(F)F)=O)CN(C(c2cnsc2)=O)CCC1C(F)(F)F C(CC(O)C(=O)NCC1CC1Cl)NC(C1(CC=C)CCCC1)=O c1(C(=O)NC2CN(C(c3c(SC)csc3)=O)CC2C)noc2c1CCCC2 c1(CC(=O)NC2CC(CCNC(c3[nH]cc(C)c3)=O)C2)ccc2c(c1)CCCO2 C#Cc1ccc(C(=O)N(CC(C)CNC(=O)Cc2ccc(Br)nc2)C)o1 Nc1ccc2nc(C(=O)NCCc3ncccc3F)ccc2c1 C1(CCNC(c2cccc(NC)c2)=O)CCN(C(c2snc(C)c2N)=O)C(C)C1 C1(N(C(CSC)=O)C)CCCC(NC(c2ncccc2-c2ccccc2)=O)C1 N1(CC(=O)NCC=C)CCC(CN(C(C2CCC(C)O2)=O)C(C)C)CC1 CC(C)(CNC(=O)NCCC1CCN(Cc2ccccc2)C1)CCC#N C1(CCNC(c2c(CC)cno2)=O)COCCN1C(c1cc(C)sn1)=O c1(OCC)ccccc1C(C)NC(N1CC(c2ncc(Br)cn2)(O)C1)=O C(CCCC(=O)NC1CCC(CNS(=O)(=O)Cc2ccoc2)CC1)NC(=O)OC C(N=c1[nH]cnc(NC2CC(C)OC(C)C2)c1C)c1c(CC)n(CCC#N)nc1 c1(C(C)=O)ccc(OCCC2(C(N3CC4C(NC(C)=O)C4C3)=O)CC2)cc1 C=CC1CCN(C(C2(O)CCN(C(c3ccnc(CC)c3)=O)C2)=O)C1 C1(C(=O)NCC(c2ccccc2)C)COC2CN(C(=O)C(O)c3ccco3)CC12 Cc1ccc2ncc(C(N3CC4(CCN4C(=O)CC4OCCOC4C)C3)=O)n2c1 CC(C)C(F)(F)CCNC(=O)C(O)CNC(=O)C(C)CC1CCCC1 C1(NC(=O)Cc2ccc(Cl)cc2)CCN(C(=O)C(O)O)CC12CCC2 C1(CC(=O)NCCCN(C(=O)C=C2CCOCC2)C)COC(C)(C)CO1 C(=O)(C1CCCc2nccn21)N(CC(C)NC(C(COC)C)=O)C C1(NC(C(C2CCC2)OC)=O)CC(NC(c2ccc(F)s2)=O)C(O)C1 C(C(=O)NCCN(C(C1CCNC1=O)=O)C1CC1)(C(C)(C)C)OC(C)(C)C c1(C(CC)NC(=O)C(=O)N(C2CCCC2)C(C)C)cccc(C)n1 C1(CNC(=O)CCc2cc[nH]n2)CN(C(c2cccc(CF)c2)=O)CCC1(F)F Cc1ccc(C)c(CCCC(=O)N2CCCC2c2cn(-c3cccnc3F)nn2)c1 C(=O)(CCCCCC(C)C)NCC(CO)NC(Cc1cc(C)cc(C)c1)=O c1(-c2ncn(C)n2)ccccc1C(=O)NCCC1CN(C(=O)C2=CCC2)CCO1 N1(CC)CCCN(C(=O)CN(CC(C)C)C(=O)CSc2ccccn2)CC1 CCC(Cc1ccccc1)N=c1[nH]c2c(c(=NC(C)CCCO)[nH]1)CCC2 O=C(C1=CCOC1)NCC1CC(NC(=O)COCCCF)C1 C1(CNC(c2c(C)cccc2)=O)CCC(C)N(C(c2ccc(C(F)F)nn2)=O)C1 CN1CCN(C(C2(O)CCC2)=O)CC1CNC(c1cnn(-c2ccccc2)n1)=O C1(CC)CCCC(N=c2[nH]c3c(c(=NCC4(C5CCC5)CC4(F)F)[nH]2)CSC3)C1 c1(C(N2CCC2CNC(C23CC(F)(C2)C3)=O)=O)cn2c(n1)CCCC2 C(CCO)(C(F)(F)F)NC(COC1CCN(C(C2(C)CCNC2=O)=O)C1)=O CC(C)(C)CCC(F)C(=O)N1CC2CC1C2NC(c1ccc(CO)s1)=O CCCC(CCC)C(=O)NCC1CCN(C(=O)CCc2ccc(N)cc2)C1(C)C N1(C(CC2(OCCC)CCCC2)=O)CC(NC(C2C3CCC2CC3)=O)CC1CO N1(C(C#CCN(C(C(C)=CC2CC2)=O)CCO)=O)CCC(C)(CCO)C1 c1(C(=O)NCCN2CCN(C(C3N(C)C(=O)CC3)=O)CC2)ccc(Cl)c(Br)c1F N1(C(CCC2(C)CCN(C(Cc3n(C)cnc3)=O)C2)=O)Cc2cncnc2C1 c1(C(=O)NCC2CCC(NC(COCCC)=O)C2)ccc2nnnn2c1 c1(CC)cc(CNC(=O)C(CNC(C2CC2(F)Cl)=O)OC)on1 c1(CNC(C2N(C(CN(CCC#C)C)=O)CC=C2)=O)ccccc1F c1(C(C)=O)ccc(CC(=O)N(CCCNC(=O)Cc2cc(C)no2)C(C)C)s1 c1(C(N(C(CNC(C(CCC)OCC)=O)C)C)=O)nc(Br)c2ccccn12 CC(C)C(C(=O)NCCC(C)CCNC(=O)COCc1cccnc1)C(C)C CC1OC2CCC1(NC(=O)CN1CC3CC3C1)C2.C12CCOC(C1)C(=O)N2 N1(C(c2cn(C)nc2C)C(=O)NCCCC(=O)OCC)CCOC(C)(C(F)F)C1 N(C1CCCc2ccc(F)cc21)(CCNC(C1C(C)CS(=O)(=O)C1)=O)C1CC1 c1(C(=O)NC2CC(C)N(C(c3cnn(CC(F)(F)F)c3)=O)C2)cnc(O)c(Cl)c1 CC1C(C)CCN1C(=O)CCCNC(c1csc(=N)[nH]1)=O Cc1cc(=NCc2cnc(-c3ccccc3)s2)[nH]c(NC2CCC(=O)NC2)n1 c1(NCCS(C(C)(C)C)=O)nc(N2CC(=O)NC(C)(C)C2)c2c(n1)CCCCC2 c1(C(N2CC(F)(CNC(C3CCc4ncnn4C3)=O)C2)=O)c[nH]c2ncccc12 N1(C(C(=Cc2cncs2)C)=O)CCN(C(C23CC(C)(C2)C3)=O)CC1C Cc1ccn(C(C)C(=O)NC2(CCCNC(=O)CCn3ccnc3)CC2)n1 C1(NC(C(C)(C)O)=O)CN(C(=O)C=Cc2ccc[nH]2)Cc2nccn2C1 C#CCC(CC(F)F)C(=O)NCC(CC)(CC)C(=O)N(C)CCc1cccnc1 C#CCC(CC#C)C(=O)NC(c1cccc(OC)c1)CNC(C1(OC)CC1)=O CC1CN(C(=O)CSc2ccccn2)CCCN1C(=O)C=CI c1(C(=O)NC(CCC)CCCNC(=O)CC(C)(C)O)scc2c1OCCO2 C1(CNC(C2CCC(CC)C2)=O)CCC(NC(c2ncoc2C)=O)CC1 C1(C2CC2)(CNC(CS(CC)=O)=O)CCN(c2snc(C)c2C#N)C1 C(=O)(C(C)CC(C)(F)F)NCC(CC)NC(C1C2CN(C)CC12)=O C1(C(C)(C)C)CC(C(=O)N2CCCN(CC(=O)NC3C4CCCC34)CC2)=NO1 c1(C(=O)NC2CCC(N(C)C(c3ccon3)=O)C2)cccc(O)c1 C(=O)(CN(C(=O)CN(C)CC1CC1OC)C)NCC=C C1(c2cn(C)nn2)OCCCC1CNC(=O)C=CCOc1ccc(Cl)cc1 C(O)(CNC1CCCN1C(c1ccc(Br)cc1I)=O)(C(F)(F)F)c1ncc(C)o1 N1(C(C2N(CCC)C(=O)CC2)=O)CCC12CN(C(=O)C(C)Cc1ccccn1)C2 C1(NC(C(C)n2cnnc2)=O)CN(C(=O)CN2CCC2)Cc2nccn2C1 c1(OC)ccc2cnc(N3CCC3(C)CNCc3ccc(Br)c(C#N)c3)nc2c1 C1(C(NOC(=O)CC2CCCOC2)=O)CN(CC2CCN(C)CC2)CCN1C c1(C(=O)NC2C(F)CCN(C(CCC(=O)N(C)C)=O)C2)cc2ccccn2c1 C=CC1(C(N2CC(OC)C2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 CCC(CNC(=O)C(O)C(C)SC)(CC)NC(c1cnn(C)c1C)=O c1(C(=O)NCCc2ccc(C)cc2Br)cccc2c1CC(=O)N2 CCN(OC)C(=O)CNC(=O)C(CCSC)NC(=O)C(N)=O N1(C(CNC(C(CC)C)=O)=O)CC(C(=O)NCc2cnc(C)cn2)C2(CC2)C1 Cc1c(C(N2CC(O)(CCNC(c3ccccn3)=O)C2)=O)cc(N)cc1O C1(NC(c2c(N)nccc2)=O)CC12CCC(NC(C1CN3CCC1CC3)=O)CC2 C1(C(=O)CCN)CCC(=O)N1.N1(CC(C)C)CC(C(=O)NC(=O)CSC)C1 C1(CC(N2CC(CNC(CC3CC(=C)C3)=O)C2)=O)COCC(C)O1 CC(C)CC(C(=O)N1CCOCC1CCO)N(C(=O)C(=O)NCC(F)F)C CC(C)(C)CC(O)C(=O)N1CCCC(CNC(c2ccn3c2CCCC3)=O)CC1 c1(C(N2C(CN(C)C(C3CSCCS3)=O)CCC2)=O)cncc(Cl)c1Cl c1(CCNC(=O)NCc2ccnc(C(F)F)n2)cc(Br)ccc1Cl C(c1cccc([N+](=O)[O-])c1)=CC(N1CC2C(NC(C3(C)CCN(C)C3)=O)(C2)C1)=O N1(C(c2c(CC)n[nH]c2)=O)CC(C2CC2C(=O)N(C(C)(C)CO)CC)C1 C1(NC(CNC(CCCCC)=O)=O)CC2(CCN(C(=O)C(C)(C)C3CCC3)C2)C1 CCC(C)(C)C(C)CC(=O)NC1CCC(NC(C2CCCCC2)=O)CC1 C1(N(C(C(CC=C)(C)C)=O)C)CCCC2CN(C(=O)C3=C(C#N)CCC3)CC12 C1(CCNC(CN(C(C)C)C(C2CC(=C3CC3)C2)=O)=O)CCCOC1 c1(C(=O)NCCC2CC(NC(c3cncc(OC)c3)=O)C2)cscc1S(C)(=O)=O n1(CC(=O)NC2C(NC(C(C(C)C)OC)=O)C2)cnc2cc(C)c(C)cc12 C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)NC(c2ncc[nH]2)C)CC(C)C1 C(CCC(=O)NCc1nc(CNC(=O)CC2(C)CC2F)cs1)N(C(C)=O)C N1(C(C2C(NC(CCC3CC(OC)C3)=O)C2C)=O)CCC(N=[N+]=[N-])C1 c1(N(CC(=O)NC2C(NC(C(c3cncnc3)C)=O)C2)C)ccc(Br)s1 C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)CC2=CCCC2)CC(F)(F)C1 c1(C(=O)NC2C(CNC(C3(CCC)CC3)=O)C2)cn(C)nc1-c1ccoc1 C(=O)(CCC(=O)NC(C1CCN(C(c2cc(C(F)(F)F)cs2)=O)CC1)C)NC C1(NC(C(C2CCC2)OCC)=O)CC2CC1CC2NC(C1(OC)CCOCC1)=O CC(C)CC(O)C(=O)NCC1C2CN(C(c3[nH][nH]c(=N)c3Br)=O)CC12 N1(C(C(C=CC)O)=O)CC2(CCC(CNC(C3CC3(F)F)=O)O2)C1 c1(C(N(C)CC2(NC(C(C(CC)C)O)=O)CC2)=O)ccc2c(c1)CCCO2 c1(C(N(CCCCCCNC(C(n2c(C)ccn2)C)=O)C)=O)ncnc(O)c1F C=CCCCCCCC(=O)NCC1CC(c2ccccc2)C1(C)C C(c1ccc(F)cc1)=CC(N1CC(C(C)NC(C2CC3(CC3)C2)=O)C1)=O Cc1c(C(=O)NC(CC(=O)O)C2CC2)cc(C2CCCC2)n1C C12(C(=O)NC3CCN(C(C)=O)CC3)COCC1CN(CCn1nccn1)C2 Cc1cc(Br)c(C(=O)OCC2(C)CC(C)C2)s1 c1(CSCC(N2C(C)CC(CNC(C(C)N(C)C)=O)C2)=O)ccc(N(C)C)cn1 C1(NC(C(C(C)C)N(C)C)=O)CC2CC(NC(=O)Cn3cc(C(N)=O)nn3)C2C1 n1(CC(N2C(C)CCC(CNC(=O)CO)C2)=O)ncc2cc(Br)cnc12 N1(CC(=O)n2c3ccc(cc3)c2=O)CC2C3C=CC(C3)C2C1.C1(CC)CCCC1 Cn1cnc2nc(=NCc3c(F)cccc3Br)[nH]c(NCCC3SCCS3)c12 c1(OC(C(=O)NCC(C)CN(C(=O)CCC(F)F)C)(C)C)ccc(F)cc1 C1(C(=O)NC2CCN(Cc3c(C)ccc(Br)c3)C2)CCc2nc[nH]c2C1 C12CN(CC13CC3)C(=O)S(=O)(=O)C2.NC1CCN(C(=O)NCCCCl)C1 N1(C(C=CC(=O)OC)=O)CCN(C(=O)C(C)c2ccco2)CC1C(C)C C(=O)(CCCS(N)(=O)=O)N1C(CNC(Cn2c(C(F)F)cc(C)n2)=O)CC2(CC2)C1 Cc1cc(C)c(C(N2CC(C(C)NC(C3COC(=O)O3)=O)C2)=O)c(S)n1 N1(C(C(=O)COc2cc(C)on2)=O)CCC(C)(CNCC)C1.c1(C(CC)OC)ncc[nH]1 c1(NC(C(CC)n2cncn2)=O)c(Cl)cc(C)nc1Cl C(c1ccc(C)o1)=CC(=O)NCC(CCNC(c1c(CC)n[nH]c1)=O)OC C1(C)(C(=O)OCC2CCN(C)CC2)COCCN(C(=O)NCC(C)(C)C)C1 Cc1cccc2c1CCC2N(C)C(=O)CC1CCS(=O)(=O)C1 c1(C(=O)NC(C(C)C)CCN(C(=O)CC2CC2)C)ccc(Cl)c(F)c1N C1(C(=O)NC2CC(NC(C3(CCCC)CC3)=O)C2)CCC(C(C)C)CC1 N1(C(CCOCC)=O)CCN2CCN(C(C3CCNC(=O)C3)=O)CC2C1 c1(N2CCN(C)C(C)(C)C2)nc(=NC2CCSCC2)[nH]c2c1SCC2 C1(C2(O)CN(C(c3cnc(C(F)F)c(F)c3)=O)C2)(CNC(CC(C=C)C)=O)CC1 C12CCCN(C1)C(=O)CCOCCON2C(=O)C1CC1.CCC c1(C(C)NC(=O)Cn2cccn2)ccc(CNC(=O)CN2CCCNC2=O)cc1 C1(C(=O)NC2CCCN(C(c3cnc(OC)s3)=O)C2)CCc2cnn(C)c2C1 O=C(CC(C(F)(F)F)N1CCOCC1)NCCC1CN(C(C2COCCO2)=O)C1 c1(C(N2CC(C)(CC(=O)NCc3c(C)cc(C)nc3)C2)=O)c[nH]c2ncccc12 C(=O)(CC(C)C(F)F)NCC=CCC(N1CCCC(CCC)C1)=O Cc1cc(CNC(=O)CC2CC(NC(=O)C(C3CC3)C3CC3)C2(C)C)cnc1F c1(OC(C(=O)NCC(CNC(CC2(C=C)CC2)=O)(C)O)CC)cccc(Cl)c1 c1(OC)cc2c(=NCCC3CCC(CO)O3)[nH]cnc2cc1F Cc1oc(C#N)cc1C(N1CCC(NC(=O)Cc2cscn2)C12CC2)=O c1(CN(CCNC(CCC=CCCC)=O)C(c2ccc(Cl)[nH]2)=O)cccc(C)c1 c1(-c2n(-c3ccn(CC)n3)nc(-c3nccs3)n2)cc(C)c(C)cc1Cl c1(OC)ccc(CCNC(C2CC2F)=O)cc1-c1nn[nH]n1 C1(COC)C2CCN(C(=O)NC(CNc3cc(C)c(C)[nH]3)C(C)C)CC12 C1(NC(c2c(CC)non2)=O)CCCC(C(=O)NN2CCCC(O)C2)C1 C1(CNC(CCOC)=O)CN(C(c2conc2-c2ccccc2)=O)CC12CCC2 c1(COC(CC(C(C)C)c2ccon2)=O)ccc2nc[nH]c2c1F C(=O)(C1=NN(C)C(=O)CC1)NC1C2(C(=O)NCC3(CC)CCOC3)CCC(C1)C2 N1(c2cc(NC)nc(COC)n2)CC(NC(C2(OC)CCC2)=O)C2CCCCC12 c1(CC(=O)NC(CC)(C)CNC(=O)C=Cc2ncc[nH]2)cc(OC)c(O)cc1F N1(C(C2(CO)CCC2)=O)CCC(F)(C(=O)Nc2ccc(CCO)cc2)C1 C#CC1CC2CCC1N(C(C1C(C(=O)NC(C)COC(C)C)C1)=O)C2 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CN(C(CC(=O)OC)=O)C(C(=O)OC)C(O)C1 c1(COC(c2c(CC)cno2)=O)ccc(N(CC(C)(C)C)C)cc1 C(CC1=CCN(C(c2ccc[n+]([O-])c2)=O)CC1)NC(=O)CC1CN2CCN1CC2 c1(C(=O)O)nscc1S(=O)(=O)N1CCC(c2ccccc2)C(O)C1 C(C)(C)(CCCNC(=O)C(c1ccc(Cl)s1)=O)NC(C1CC(SC)C1)=O c1(CN(CCCC2CCOC2)C)cc(Cl)sc1Cl Cc1cc(C(=O)NCCN2CCCN(C(=O)C(C#N)C3CC3)CC2)cc(F)c1C S(=O)(=O)(CC(=O)NCCCC1CCCCN1C(C1CC(C)=NO1)=O)NC N1(C(c2cn(C)nc2)=O)CC(NC(=O)Cc2c[nH]ccc2=O)CC12CCCC2 N1(C(N=c2ccn(C)[nH]2)=O)CC2OCc3cnnn3C2C1.c1ccncn1 C1(NC(CC2(OC)CCCC2)=O)CCC(C)(CNC(=O)C(F)=C(C)C)C1 CC1(C(=O)NC2CN(C(c3ccc(=O)oc3)=O)CC2n2cccn2)CC2CC2C1 C(C(C(=O)NCC(C)C)N(C(C)C(C)C)C1CC1)C1CC(C(=O)OC)C1 C(CC(C(=O)N1CCC1(C)C(=O)NC)NC(=O)CC1CC1C1CC1)=CC N1(C(=O)Cn2cccn2)CCN(C2CCN(C(c3cc(Br)c[nH]3)=O)C2)CC1 c1(C(C)C)ccc(C(=O)N(C(c2ccccc2)CO)CCO)nc1 C(=O)(CCCF)NC(C1(C(=O)NC(c2ccsc2)C)CC1)C c1(C(=O)NC2C(CC)CN(C(C3CC(C)(C)C3)=O)CC2)cccc(Cl)c1[N+](=O)[O-] N1(C(Cn2c(C)nnn2)=O)CCC(C(=O)NCC2(C)CCCO2)C(O)C1 c1(NCCC2CCN(C(c3ccnc(O)c3Br)=O)C2)ncccc1[N+](=O)[O-] c1(C(=O)NC2C(OC)CN(C(c3ncn(CC)n3)=O)C2)nnn2c1CSCC2 Cc1ccc(F)cc1C(N1CCC(C)C(CC(N2C3COCC2C3)=O)C1)=O c1(OC)cc(C(N2CCOCC(NC(=O)C3=CCOC3)C2)=O)c(Cl)cn1 N1(CC(=O)NC2CC(NC(=O)CC3CC3)C2)C(=O)C2C3C=CC(C3)C2C1=O CC1CCN(C(C2(CNc3cc(C(N)=O)[nH]n3)CC2)=O)CC1CO C(=O)(C(CC)C(=O)NCc1nc(CNC(c2[nH]ccc2COC)=O)cs1)OCC C(=O)(C1=CCCOCC1)NC(c1cn(C)nn1)C(N1CC(C)(C)CCC1CNC)=O c1(N2CCCC(NC(C3C(CC)CCC3)=O)CC2)nc2cc(F)ccc2o1 c1(CCC(N2C(CNC(C3(C)C(C)C3)=O)C(O)C(O)C2)=O)c[nH]c2ccccc12 c1(C(=O)NCC2(OC)CCN(C(=O)Cc3c[nH]nc3C)C2)nc[nH]c2nccc1-2 c1(OC)cc(Cl)cc(C(C)CCN2CCN(C(C3CC(=O)N(C)C3)=O)CC2)c1O C1(NC(C2CCCC(F)C2)=O)CCC2CN(C(=O)CCCCC3CC3)CC2C1 C(=O)(C1=CCCN(C(c2cccn(C)c2=O)=O)C1)NC(C#C)C C1(NC(c2c(C)con2)=O)CCN(C(C2CC(C)(F)C2)=O)C(C)C1 CC1(C)CCC(C(=O)NCCCN(C(=O)CCCC2CC2)C2CC2)c2ccccc21 N1(C(C2CCOC2)=O)CCOC2(CCN(C(C34CC5CC3(CO)CC5C4)=O)C2)C1 N1(C(c2onc(CC)n2)=O)CCC2CC2(NC(c2ccnnc2C)=O)CC1 N1(C(CC=C)=O)CCC(C)C1CNC(c1cnc(Cc2ccsc2)s1)=O C1(C(N(CC)CC2CCCCN2C(=O)CCN2CCC2)=O)CC2C(C1)C2(C)C C(=O)(C1CCc2nccn21)N1CCC(CNC(c2c(CC)ncs2)=O)C1 Cc1c(C(N2CCC3CC23C(=O)NCc2cccnc2)=O)[nH]ccc1=O C1(NC(C(C)C2CCOC2)=O)CC2(CCN(C(=O)C3=CCCC3)CC2)C1 c1(C(N2C(C)C(NC(=O)C(Cl)=CCl)CCC2)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(C(CC)(F)F)=O)CC(NC(=O)Cc2ccc(F)cc2)C2(CCCC2)C1 C12(C(N3C(C)(C(=O)OC)CCC3)=O)CCC(CN(C(=O)C=C(C)C(F)F)C1)C2 c1(OCC(=O)NC2CCC(NC(C3C(=C)CC3)=O)C2)ccc(C(C)=O)cc1CC C#CC1CCCCN1CCC(=O)NC1CCCN(Cc2ccccc2)C1 C1(NC(CC(C)OC)=O)CN(C(c2ccc(C(C)C)cc2O)=O)CCC1C C#CCC(C)(C(=O)N(C1CC1)C(C)C1CC1)NC(c1cccc(OC)n1)=O C1(C(N2CC(NC(c3n(C=C)ncc3)=O)C(C)C2)=O)CCc2nn(C)cc2C1 N1(C(C2N(C(C)=O)CC3CC32)=O)CC2(C1)CN(C(C1CC3(CCC3O)C1)=O)C2 CC1CCc2onc(C(=O)NCC3CC34CCCCCC4)c2C1 c1(C(=O)NC(CN(C(c2c(SC)cc(C)cc2)=O)C)C)cnn2c1CCCC2C C1(C(=O)NC2CC(NC(COCCC)=O)C2)CCC(NC(C)=O)C1 c1(OC)ccc(C(N2CC3(CC3C(=O)NC(C3(O)CC3)C)C2)=O)c(OC(C)C)c1 c1(CC(=O)NC2(C(C)NC(=O)Cc3ccc(F)cc3)CC2)c(C)cccc1Br CC(C)C(C#N)C(=O)N(C1C2CN(C(=O)Cc3nc(C4CC4)cs3)CC12)C c1(C(=O)Nc2c(C)cc(NC(=O)CCOCC(C)C)cc2)nn(C)c2c1CCC2 Cc1ncccc1C=CC(=O)NCC(C)(C(C)C)NC(=O)CN1CCC(C)C1 c1(C(=O)NC(CC)CNC(c2ccc(OC)cc2O)=O)ccc2c(c1F)CCC2 C1(C(C(=O)NCCOC)N(CCN(C)C)Cc2[nH]cnc2C)CCC(C)(C)CC1 CCS(=O)(=O)CC(=O)N1CCC1CNC(C1CCC(n2ccnn2)CC1)=O Cc1ccc(SCC(=O)NCCCN(C)C(C2CC3(C2)CC3F)=O)cc1C C1(CNC(c2cnc(C(F)(F)F)cn2)=O)CCC2(CCC2)O1.CC1CC2CN1C2 C(C(O)CCNC(c1cnoc1-c1ccco1)=O)NC(C1(C(N)=O)CC1)=O c1(C(=O)NC2CC(CNC(c3cccnc3C3CC3)=O)C2)ccc2nn[nH]c2c1 C(CC(=O)NCCOC(C)C)(C(C)C)NC(c1cc(C)sc1C)=O C1(NC(=O)CCC2CC2)CC12CCC(NC(c1ccc(CO)cc1F)=O)CC2 C(C(=O)NCC(C)S(C)(=O)=O)(C(C)C)NC(c1c(CC)nns1)=O c1(C(=O)NCCCC(C)NC(c2c(C)onc2C2CC2)=O)nc(O)[nH]c(=O)n1 c1(C(=O)NC2CCN(C(c3cccc(C)c3O)=O)CC2O)ccc2nc[nH]c2c1 CC1(C)NC(=O)CC1C(=O)NCC(CO)NC(=O)Cc1c(F)cccc1Cl CCC(C)(CNC(C1CCN(C(=O)C=CC2CCC2)CC1C)=O)C(N)=O N1(C(CCCCC)=O)CCN(C(c2cnn(C3CCCC3)c2C)=O)CC1CO C1(C(N2CCC(OCCC)CC2)=O)CCC(CC)NC1=O C1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)ccn2)=O)COC2COCC12 N1(C(CCC=CCC=C)=O)CCC(F)(C(N2CC(C)CC(O)C2)=O)CC1 c1(C(=O)NCC(CNC(C=CCOC)=O)CO)cccc(OCCF)c1.S(C)(=O)(=O)N c1(NC)ccccc1.C1(NC)CC(NC(C2(CC(=O)N)CC2)=O)CC1O.CSCSC N1(C(c2ccn(C)c(=O)c2)C(=O)NCCC)CCCN(C)CC1C c1(CC)nc(C(=O)NCC2CCN2C(C2CCCC2OC)=O)cs1 c1(C(=O)NCC(CNC(c2ccc(C(=O)OC)s2)=O)F)cc(Cl)nnc1O N1(C(C(C)NC(=O)NCCC(=O)N(C)C)=O)CCCC2(CCCCO2)C1 C1(CNC(c2c(CC)cno2)=O)C(C)CCN1C(c1cc[nH]c(=N)n1)=O Cc1ccc(C(=O)N(CC(C)O)CCN)n1C.C1(C(=O)NC(C)C)CCCN1C(C)C N1(C(C2(OC)CCCOC2)=O)CC(C2CCN(C(C3C=C(C)CS3)=O)CC2)C1 C1(CNC(C2(NC(c3ccc(C)o3)=O)CC(F)(F)C2)=O)CC(C(N)=O)=NO1 N(C1CCCn2ccnc21)C(=O)CC1(CO)CC1.C1(=O)C(O)CN1C1CC1 C#Cc1ccc(F)c(C(N2CC3CCC2(CNC(=O)CC(C)CCC)C3)=O)c1 N1(Cc2ccc(C)s2)C(=O)NC(CC2(C)CC2)C1=O CC12CN(C(=O)Cn3cc(Cl)cn3)C(C(=O)NCC3CC3c3ccoc3)(C1)C2 c1(N)ncc(C(F)F)cn1.C1(C(C)=CCNC(=O)C2CC2)(COC)CC1 N1(C(CC#N)=O)CCC2CN(C(c3cc(-c4ccccc4)[nH]n3)=O)CCC12 c1(CC)cc(OC)ccc1C(=O)NCC1CC1NC(=O)C(C)Cn1cccn1 N1(C(C(CCSC)NC(CCC)=O)=O)CC2(C1)CN(C)C2 C1(OCC)CC2(C1)CC2C(=O)NCC1CC(C)N(C(c2cnn(CC)c2)=O)C1 CC1=NNC(=O)C1CCC(N1CC2CC2(CNC(C2(C)CC(F)C2)=O)C1)=O C1(C(C)C)CN(C(=O)C(O)C(C)C)CCN1C(c1cc(C(N)=O)cn1C)=O Cc1cnncc1C(=O)NC1(CN(C)C(c2ccc(N(C)C)nc2)=O)CC1 O=S(=O)(c1cccc(=NCC23COC(CCO2)C3)[nH]1)NCCC=CBr Cc1cc(=NCC2(C(C)(C)C)CC2)[nH]c(N2CCC(COC(C)(C)C)C2)n1 CC(O)(CNC(=O)CC1CC2(C1)CN(C(c1cnncc1O)=O)C2)C(F)(F)F C=CC1COCC1NC(C1(C(C)NC(C2(O)CCC2)=O)CC1)=O Cc1cccc2c1CC(C(N1CCC3CCN(C(=O)CSC(F)F)CC13)=O)O2 C1(CC2CC2)CCN(C(c2c(NC(N)=O)cccc2)=O)C(c2ccncc2)C1 c1(-n2ncc(C(=O)NCC(C)(CO)NC(C3C(OCC)C3)=O)c2)cc(C)ccn1 c1(CN=c2scc(CN(C)C)[nH]2)ccc2c(=O)cc[nH]c2c1 Cc1cc(C(=O)NCC(C)(C)OCCNC(c2cncnc2C2CC2)=O)c(C)s1 CCC(CNC(=O)C=Cc1cnc(C)s1)(CC)NC(c1ccn(C2CC2)c1C)=O c1(C(=O)NCCNC(c2cncc(OC(F)F)c2)=O)cc(Cl)c2ccncc2n1 N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CCC(NC(=O)CC(C)C(C)C)C(O)C1 c1(C(=O)NC(CNC(c2c(CC)ccs2)=O)CO)cc(C)ncn1 N1(C(c2c(C(C)C)onc2)=O)CC2(CCN(C(=O)CCCN3CCCC3)CC2)C1 c1(C(=O)NCC2(F)CCC(CNC(c3ccncn3)=O)C2)ccc2sccc2c1 c1(C(=O)NCCN(C(C(C)CC2CCCC2)=O)C2CC2)csc2cccnc12 c1(C(N2CC(NC(c3cncc(C)c3)=O)C(F)C2)=O)ccc([N+](=O)[O-])cc1Br c1(C(=O)NC2(C)CC(NC(Cn3c(C)nnn3)=O)C2)[nH]cc2c1CCS2(=O)=O C1(CC(=O)NCCC2CCN(C(C34CCC(CC3)C4)=O)C2)CCCS(=O)(=O)C1 N1(C(COC)=O)CCN(C(=O)CSC)CC1c1cn(Cc2cccs2)nn1 N1(C(C2C(C)C2C)=O)CCC(OC2CN(C(=O)CCCCN3CCOCC3)C2)CC1 C1(NC(=O)NCC(N2CCN(C)CC2)C)C(C)(C)C(NC(=O)OC(C)(C)C)C1(C)C C1(CC(=O)NC(CNC(C(CC)C)=O)(C)C)CCN(C)C1=O n1(CCNC(C2C(C)C2C)=O)cc(C(N2CC(N3CCCC3)C2)=O)cn1 C(C)(CC(=O)NCC1CCN(C(c2cc(C3CCC3)[nH]n2)=O)C1)SC Cc1ccn2cc(C(=O)NC(C)(C)CCNC(=O)C(C)(F)C(F)(F)F)nc2c1 C1(CNC(C(C)O)=O)C2CC1CN(C(=O)CONC(=O)OC(C)(C)C)C2 CCCCCCC(=O)NC(C)(C)CN(C)C(c1cc(Cl)cnc1O)=O Cc1cc(O)c(C(N2CCN(C)C(CNC(C3CC34CC(F)(F)C4)=O)C2)=O)nn1 C(CC(C)C(=O)N(C)CC1CN(C(=O)C(=O)NCC2CC2)C1)=CCC C#Cc1cn(C)nc1C(N1CCCC(O)(CCNC(c2[nH]cnc2CC)=O)C1)=O N1(C(C2CC(C)OCC2)=O)CC2(C1)CN(C(=O)CCC1CCCC1)CC(C)(C)O2 C(=O)(C(C)(F)C(C)(C)F)N1C(CCNC(C2=C(C)CC2)=O)CCCC1 C1(CC(=O)NC(C2CCN(C(=O)CC3(C#N)CC3)C2)C)SC2=NCCN2C1=O Cc1o[nH]c(=NC(=O)NCCC2CCC(=O)N2)c1C C1(NC(C(CCC)CC)=O)CCCCCN(C(=O)CSc2cn[nH]c2)C1 c1(CN2CCC(NC(c3cc(Br)cc(Br)c3)=O)C(O)C2)c(Br)ccc2c1OCO2 CC1CN(C(=O)CC2CCCCO2)CC1NC(=O)CC1C=CCC1 CCS(=O)(=O)CC(=O)N1CCCCCC1CNC(c1cc(O)nc(O)n1)=O c1(C(=O)NCC2(O)CN(C(C(C3CC3)OCC)=O)C2)c(C)n[nH]c1C c1(OCC)nc(NC2CN(C(=O)CN3CCNC(=O)C3)C2)nc2ncn(C)c12 N12CCCN(CC1)C(=O)C2.C1(=CC(N2CCC(OC)C2)=O)CCC(C)(C)CC1 c1(OC)ccc(OC)c(C(=O)NCCC2CCC(NC(=O)C(C)=C3CCC3)C2)c1 N1(C(c2ccc(C)cc2C)C(=O)NCC(F)F)CC2(CCOCC2)C1CC(C)C C=CC(CCC)CC(=O)NC1CCC(CCC(=O)Nc2ccccc2C)C1 C=CCCC(F)(F)C(=O)NCC(C1CCN(C(=O)C(F)CN(CC)CC)CC1)C C(C(C)(C(C)C)NC(c1cccc(NC(=O)OC)c1)=O)NC(C1C(=C)CC1)=O c1(OC)cc(C(=O)NC(c2cscn2)C)c(NC(C2CC2C(N)=O)=O)cn1 C1(C(=O)NC2CC3(CN(C(C=CCC)=O)C3)C2)CC2CCCCC2O1 c1(NC2CCCCN(C(c3cnn(CCO)c3)=O)C2)nccn2nnnc12 N1(C(C(CCC)=CCC)=O)CC23CCCC2(C1)CN(C(C1CCOC1CC)=O)C3 C(=O)(C1=NOC2COCC12)NCC(=C)CCNC(c1cc2cccnn2n1)=O c1(C(=O)NC2C(NC(C(C)Cc3ccccc3)=O)CCC2)cc(N)cc(O)c1F c1(C(=O)NC(CN(C(Cc2cc(C)on2)=O)C)C)noc(Cl)c1Br Cc1c(C(N2CCN(S(=O)(=O)CCCl)CCC2C)=O)cc(F)cc1Cl c12cc(sn1)C=CC(=O)N2C.C1(N)CCC(CNC(=O)CSCC(N)=O)C1.CO CN1CC=C(C(=O)NC2CCC(CNC(=O)COCc3nc[nH]n3)C2)C1 C1(C2CN(C(=O)Cc3cncs3)C2)(NC(C(C)OCc2ccc(C)cc2)=O)CC1 N1(C(C(C(CC)O)C)=O)CC(NC(=O)Cn2cnc(C(F)(F)F)c2)C2(CCC2)C1 c1(CC=C(C)C)ccccc1C(=O)N(CCCNC(C1CCCO1)=O)C C(=O)(CC1=CCCC1)OCC(c1n(CC=C)nnn1)NC1C(CO)C2CCCC12 c1(C(=O)NC(C(C)NC(c2c(CC)c[nH]n2)=O)(C)C)cn(C)c2ccc(F)cc12 N1(Cc2occ(C(=O)OC)n2)CCN(C(C2CC(N(C)C)C2)=O)CC1 C12(C(=O)NC3C4CN(C(C5(N(C)C)CCC5)=O)C3C4)CCC(C)(C1)OC2 C1(CC(=O)NC(C(N)=O)=O)(NCc2[nH]ccc2C2CC2)CCOC1 c1(C(N2CCC(NC(C3CCC(COC)C3)=O)C(O)C2)=O)cc2oc(C)cc2[nH]1 C1(C(=O)NCC2(COC)CN(C(C3(CO)CCCCO3)=O)C2)CC(=O)N(C)C1.C1CC1 C1(=O)C(C(CC)CC)Oc2c(CN3CC4(CC4)CC3CC)nsc2CN1.O(C)CC C1(C(N(C)CC2CCCCN2C(=O)Cc2cc(Cl)cs2)=O)CCc2nnnn2C1 CCC(CC)CCC(=O)NC1CC(C)N(C(c2ccc(S(C)(=O)=O)[nH]2)=O)C1 C1(OCC(=O)OC)CCN(C(c2csc(C)c2)=O)C1 Cc1c(C2OCCC2C(=O)NCCN(C(=O)CC2CN(C)C2)C2CC2)cnn1C N1(C(C=CCOC)=O)CCC2CCC(NC(c3cc(C)c(C)c(C)c3)=O)C1C2 c1(C(N2CCC(N(C(C(F)=CCC)=O)C)CC2)=O)cc(Cl)cc(Br)c1 N1(C(C(C)(C)OC(C)=O)=O)CCC(O)C(NC(C2(C(F)(F)F)CCCC2)=O)C1 N1(C(C2(CC)COC2)=O)CCn2nc(C(=O)Nc3cccc(O)c3)cc2C1 c1(CC(=O)NC(C)CCNC(C2CN(C)C(=O)N2)=O)cccc2cccnc12 N1(C(CNC(=O)CNC(C2(O)CCCCC2)=O)=O)CCOC(CO)C1 CC1CC(NC(=O)CCc2cn[nH]c2)CN1C(=O)COC1CC1 C1(C(=O)NC2CN(C(C(C3CCCCC3)C)=O)C2)CCC2CC1C2(C)C N1(C(C(COC)C)=O)CC2(CCCCC2NC(c2cn(C)c(=O)nc2O)=O)C1 C1(CNC(=O)C(O)CC2CC2)CCCN(C(c2cnn(-c3nccs3)c2)=O)CC1 N12C3CCC1CN(C3)C(=O)CC2=O.CCC(CC)(C(F)(F)F)c1ccccc1 C1(C(=O)NC(C(=O)N(C(C2CCCO2)C)CC)CCSC)CCC2(CC1)CC2 C1(C)(C(=O)NCC=CC(N2CC=CC(OC)C2)=O)CCCN(C)C1 C1(C(=O)NC2CN(C(C3CCN3C3CCCC3)=O)C2)(CC)CCOCC1 N1(C(C(CCSC)O)=O)CCC2(CCC2NC(c2cc3ccccc3[nH]2)=O)CC1 C#CCCC(O)C(=O)NC1COCC1CNC(c1c[nH]c(=O)cn1)=O c1(OC)ccccc1-n1cc(C2(C)CN(C(=O)COc3ccc(Cl)cc3)C2)nn1 N1(C(C(=Cc2cccs2)C)=O)CCC(C(C)(C)NC(C2COC(C)C2)=O)CC1 C1(CNC(Cc2c(C)occ2)=O)C(C)CCN1C(c1ccnc(O)c1)=O c1(-c2n(CCCCC)nc(C3CCCO3)n2)sc2[nH]c(C)nc(=O)c2c1C N1(C(C=C2C(C)(C)CCCC2)=O)CCC2CC2(NC(=O)CCCN2CCC2)CC1 Cc1cc(=NC2CC(CNCCO)C2)cc(C)[nH]1 c1(N2CCC(NC(C=CC=CCC)=O)CC2C)ncnc2n[nH]cc12 C(=O)(CCN(OC)C(=O)CN(CC(C)CC)C)NC(C=C)COC N1(C(c2n(CC)cnn2)=O)CCC(C)C(NC(C2CCN(CC3CC3)CC2)=O)C1 c1(C(=O)NCn2cnc(C(=O)OCC(C)C)n2)cn2c(n1)CCC2 N1(C(CS(CC)=O)=O)CC(NC(c2cccc3c2CCO3)=O)CC12CCCCC2 c1(C(N2CCC3C(NC(c4c(CC)oc(C)c4)=O)C32)=O)cc2ccc(Br)cc2[nH]1 c1(N(CC(F)(F)F)CCOC)cc(C)c(S(=O)(=O)NC2CN(C)NC2=O)cn1 S1(=O)(=O)c2ccc(c(F)c2)N1.C1(N2CCC(COC)CC2)CS(=O)(=O)CC1OC C1(CNC(c2ccc(O)nc2)=O)CC2CCC1N2C(c1csc2nnsc12)=O C1(CNC(c2cn(C)nn2)=O)CCCCCN1C(C1CCOC(C)(C)C1)=O C1(C2CN(C(C=CC(=O)NC3CC3)=O)C2)(NC(C2CC23CCC3)=O)CC1 c1(C(N(CC(C)N(C(=O)CC2CC(=O)C2)C2CC2)C)=O)ccoc1 c12ccc(s1)C(=O)NC1CCC(C1)C(=O)NC2=O.C1(CC2CC2)CC(CO)CO1.COC C1(NC(=O)C(CO)c2ccccc2)CC(F)CN(C(c2cnc(CO)nc2)=O)C1 C(C(CC=C)C(=O)NCC1=NOC(C)C1)NC(C(C=C)O)=O c1(C(=O)NCCN2CCNC2=O)nc(-c2cccnc2F)c2ccccn12 C1(NC(C2(COC)CCC2)=O)CN(C(c2ncc(C)cn2)=O)CC1O C12(C(N(CCCNC(C=C(C)c3cccs3)=O)C3CC3)=O)CCC(C1)C(C)O2 C(N=c1ccnc(C2CCC2)[nH]1)C1CN(C(Cc2ccn(CCOC)n2)=O)C1 N1(C(C(C2CCC2)OC)=O)CCC2(C1)CN(C(c1cc3c([nH]1)CCCC3)=O)C2 c1(CC(C)NC(C2=CCSC2)c2n(CCC)nnn2)ccc2c(c1)CCC2 Cc1cccc(C(=O)NCC2(C(N3CC(F)C3)=O)CC(C)(C)C2)c1N C1(CNC(C(C)SCC)=O)CC2CCC1N2C(c1cc(F)cc(F)c1)=O c1(C(N2CCC(N(C(=O)CSCC(N)=O)CC)C2)=O)c(C)ccc(F)c1N C(CC(=O)NC(C)(C)C)(C(F)(F)F)NC(C(c1cccc(C)c1)O)=O.C1(C)CC1 C(Cn1cncn1)(C(=O)NC1COCC1O)NC(c1sccc1Cl)=O C12(C(=O)NC(CCNC(CCCNC(C)=O)=O)(C)C)CCCC(=O)N1CCC2 C1(Nc2ccnc(OCC(=O)NCCOC)n2)CCNC(=O)CC1 C(c1ccco1)=CC(=O)NCC(CC)NC(c1ccc(C(=O)N(C)CC)s1)=O Cn1cnc2cccc(C(N3CCCC(NC(c4cnc(S)[nH]4)=O)C(F)C3)=O)c12 N1(C(C(F)=CCC)=O)CCC2(CC2)CC1C(=O)Nc1ccc(F)cc1O c1(C(=O)OC)ccnc(N2CCC(NC(=O)CC(C)(C)Cl)C(C)C2)c1[N+](=O)[O-] c1(C(=O)NC2CCC(CNC(c3c(C)oc(CO)c3)=O)C2)cc2scc(Cl)c2[nH]1 C1(COC)CN(C(=O)CSCC(=O)OC)CCN1C(=O)CC1CCCOC1 CC(C(=O)NC(C)(C)C)(c1nn[nH]n1)NCCC1(CN2CCCC2=O)CCCC1 Cc1ccccc1C=CC(=O)NC1CCN(C2CCCC2(C)O)C(C)C1 c1(OCC#N)cccc(NC2(c3nnnn3C3CCOCC3)CCCOC2)c1 CC1OCCCC1C(=O)NCC1CCOC1C(=O)NCCN=S(C)(C)=O c1(COC)ccnc(CNC(=O)C(C)(C2CC2)N(C)C(c2ccc(C#N)s2)=O)c1 c1(C(N2CCC(N(C(c3cc(SCC)ncc3)=O)C)C2)=O)cc(C)ccc1F C1(CC(=O)NC2CC(C)N(C(c3ccncc3F)=O)CC2)CCCC2(CCC2)O1 C(=O)(CC(F)(F)C(F)F)NC1CN(C(c2cn(CCC)nc2)=O)C(CC)(CC)C1 c1(OC)ccc(C)c(-c2cnn(C)c2CN2CCCC(c3ncccn3)C2)c1 N1(C(COC2(C)CCCC2)=O)CC2CCC1C(NC(c1cc(Cl)ccc1N)=O)C2 N1(C(c2c(OC)c(Cl)ncc2)=O)CCC2(C1)CN(C(=O)CCF)CCO2 C(=O)(C1CCC(=O)c2ccccc21)NC1CC(NC(CCC(C)(C)F)=O)C1 c1(NCCCCc2c(F)cccc2)cc(=NC2CCC2C2CCCC2)[nH]c(C(F)F)n1 c1(OC)ccc(C(N2CCC(NC(=O)C(O)C3CC3)C2C(C)(C)C)=O)cn1 c1(CSCCCNC(c2cc(C3CC3)[nH]n2)=O)cccc(C(F)(F)F)n1 CCCC(C(=O)N1CCCCCC(NC(c2cc(Cl)cn2C)=O)C1)S(N)(=O)=O N1(C(COCCOCCOC)=O)CC(NC(c2cccc(F)c2C)=O)CC1(C)C N1(C(C(C)CC#N)=O)CCCCCCC1C(=O)NCCN=S(C)(C)=O C1(C)CC(F)(C(=O)OC(C)(C)C)C(=O)N1.CCCCCCNC=O c1(C(=O)NC(C(C(C)C)NC(=O)C(c2ccccc2)=O)C)cc2ccnn2cn1 C1(NC(C(CCNC(Cc2cc(C)no2)=O)OC)=O)C(=O)NCCC1C c1(C(CC)C)nc(N(C2CCN(CCOC)CC2)C)cc(C)n1 N1(C(C(n2ncc(C)c2)C)=O)CCC2CC2(C(=O)NCCc2csc(C)n2)CC1 C12(CNC(C34CC(NC(CC5N(C)CC=CC5)=O)(C3)C4)=O)CCCN(CC1)C2 S(=O)(=O)(CCC(=O)NC12CC(C1)N(C(c1cnc(CC(C)C)s1)=O)C2)NC c1(C(C(=O)NCC2(NC(CC3C(CC)C3)=O)CCC2)O)ccc(Cl)c(Cl)c1 C1(CC)(CNC(C2CC(F)(F)C2)=O)CN(C(C2CC2C2CCCOC2)=O)C1 C123CC(C1)C(CO2)CN3.C1(C(=O)NC(C2CC2C(=O)OC)=O)(CC)CCOCC1 c1(C(N2CC(C(C)NC(c3c(C)sc(Cl)n3)=O)C2)=O)c(C)nc(C2CC2)nc1S C1(NC(CCCC(=C)C)=O)CCC(C)(C)CC1CNC(=O)C=CCOCCOC c1(NCC(N2CCC3(NC(=O)C4CC4)C(C2)C3)=O)ncnc2c1CCC2 C1(N(C(=O)CSCC#N)CC#C)CCN(C(=O)C(C)C2CC2C)CC1 CONCCCN1CCC1CC(=O)NC N=c1nc(N2CCOC3(COC(=O)NC3)C2)[nH]c(=NC2CCNC3(CCC3)C2)[nH]1 C1(CC)CN(C(=O)CC2(C)CCCCC2)CCN1C(c1cc(Br)n(C)c1)=O Cc1nsc(C)c1C(N1CCCC(CNC(=O)CC2COCCOC2)C1)=O c1(C(=O)NC2C=CCN(C(C3(OC)CCCC3)=O)C2)ccc2[nH]ccc2n1 C(CC(C(=O)NCCN1CCCOC1=O)NC(C1CCC1C)=O)OC C#CCC(CC#C)C(=O)NC1(NC(=O)C2=CCCOC2)CCCCC1C C1(COC)CN(C(C2CCC(C(N)=O)O2)=O)CCN1C(=O)Cc1sc(C)cc1C C(CC(=O)NCCC1CCOC1(C)C)(C(F)F)NC(c1c(CC)cccc1)=O c1(C2C(NCCNC(C3OCCN(OCC)C3)=O)CCC2)ccc(F)c(F)c1 c1(C(=O)NCc2ncc(C)o2)cc2c(C)cc(C)c(C)c2[nH]1 C12(CC)CN(C(=O)COc3ccccc3OC)C(CNC(=O)CC3(C)CC3)(C1)C2 C1(C(N2CC(CNC(c3sc(C)c(Br)n3)=O)C2)=O)CCOC(C)(C)C1 c1(C(N2CCCC(C(F)F)C2)C(=O)NCC=C)nc(C)c(C)n1C C(=O)(CC(C)N1CCCC1=O)N1CC(N(C(CC2(C(=O)OCC)CCC2)=O)C)C1 N1(C(C2C(C(C)(F)F)C2)=O)CC=CC1(C)C(=O)N(C1CC1)CC1(O)CCC1 N1(C(CC2CC(=C)C2)=O)CCN(C(=O)CC2CCOC2=O)C2CCCC12 CCCC(C)(C)CC(=O)NC(C)(CNC(c1cc(OC)ncn1)=O)CC(C)C c1(C(=O)NCC2(CN)CCC2)cnccc1C(c1c(CC)occ1)=O.C(F)F C1(C(=O)Nc2nnc(C(=O)NC)s2)CN(C(C(Cc2ccccc2)CC)=O)CCO1 C1(C(C)C)CCC(C(N2CCC2CNC(=O)CSc2ccccc2)=O)C(=O)N1 C1(NC(N2CCC(O)(COCCO)C2)=O)CCCOC1c1ccc(F)cc1 CC(C)C(O)C(=O)N1CCC(CCNC(c2cccc(C3(F)COC3)c2)=O)C1 N(C1c2ccccc2CC1NCC(=O)OC)C(C(=O)NC(CC)C)=O C(=O)(CC(C)CC(C)C)N1CC(C(=O)Nc2cscc2C)(SC)C1 C1(CNC(C(C2CC2)OCC)=O)CCN(C(C2(F)CCCCC2)=O)CCC1(F)F n1(COC)cc(C(=O)NCc2cc(C(N3CC4CC4C3)=O)n[nH]2)cn1 C(=O)(C1CCCc2ncccc21)NCCN(C(Cc1nc(C)oc1)=O)C1CC1 C1(OC)CN(C(=O)C=CC2(C)COC2)C(C)(CNC(=O)CCCCSC)C1 n1(C(C(=O)N(CC(CC)NC(C2(n3cccn3)CCC2)=O)C)C)cc(C)cn1 c1(NC(C2CCN(C(C(CCC)CCC)=O)C2)C)ncc([N+](=O)[O-])cc1F CC1CNc2c(CNC3CC(C(=O)NCc4ncccc4C4CC4)C3)cnn2C1 c1(C(=O)NCCC2(CNC(C3C(C)C3C)=O)CC2)cn(C2CCOC2)cn1 C1(NC(C=Cc2n(C)ncc2)=O)CN(C(c2cccc(C#N)c2)=O)C2CCCC12 c1(C(N2CC(C)(O)C2)=O)noc2c1CC(NC(=O)CN1C(=O)CSC1=S)CC2 c1(CC(=O)N(C(C(=O)N(C)C)Cc2ccccc2)C)ccc(S(C)=O)cc1 CC1(C)C2CN(C(C3CC4(CC(NC(c5cc6n(n5)CCC6)=O)C4)C3)=O)CC12 N1(C(c2c(C)oc(Cl)n2)=O)CCc2sccc2C1CNC(=O)COc1ccsn1 C1(C(=O)NCC=CC(N2CC(NC(=O)NC)C2)=O)CCCCNC1=O Cn1cc(C(=O)NCC2(CNC(=O)Cc3nccn3C)CC2(F)F)c(=N)[nH]1 C1(C(N(CCCNC(c2cnc(OC)nc2)=O)CCO)=O)CN2CCN1CC2 c1(C(=O)NCC(C)NC(=O)CSCCC(F)(F)F)c[nH]c(=O)c2ccnn12 Cn1cc(C(C(=O)Nc2ncc[nH]2)NC(=O)CNC(=O)C2CC2)nn1 C#CC1(C)COCCN1CC(=O)NCCCSn1cc(C)cn1 N1(C(COCCCC)=O)CCCC(CCC(N2CCCC2(C)COC)=O)C1 N1(C(C2(C#N)CCOC2)=O)CC2OCCN(C(=O)C3CC3)C2C1 C(C1c2ccccc2CCN1C(=O)CC(F)F)NC(c1ccc(COC)o1)=O N1(C(Cc2cc(C(C)C)no2)=O)CC2CC(C1)C2NC(c1cccc[n+]1[O-])=O C(CC(=O)NCc1ccccc1OC1CCCC1)(C(C)C)OCC O=C(CC(C(F)(F)F)NC(=O)CN1C(=O)CNC1=O)NCC1CCC=CO1 n1(CC)ncc2c1CC(C(=O)NC1CCCC1NC(=O)Cc1nonc1C)CC2 c1(C(N(C)CC2CCCC(NC(COCC=C)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(NC(c2nncc(C(=O)OC(C)(C)C)c2)=O)CCN2CCC1C2 C(=O)(C(C)(F)CO)NCC(=O)NCC(=O)NCC(COC)(C)C N1(C(CS(CC)(=O)=O)=O)CCCN(C(=O)C(F)C(C)(C)O)C(C)C1 c1(CC(N2CC(=C(F)CNC(=O)C(N3CCCC3)C3CC3)C2)=O)cnsc1 CCC(C)C(C(=O)NC(CO)C(=O)NCc1ccc(F)cn1)N(C)C C1(OC)CC(C(=O)NC(C(=O)N(C(C)CN(C)C)C)C2CC2)C1 C1(CNC(CC2N(C(C3COC(=O)C3)=O)CCC2)=O)CCC2(CCC2)O1 Cc1cn2c(CN(C)CC3CCCN3C(c3cc[nH]c(=N)c3)=O)c(C)nc2s1 c1(C(N2C(C3(O)CN(C(=O)C=Cc4cnc[nH]4)C3)CCC2)=O)cc(F)ccc1F N1(CCC2(OCC)CCC2)CC2CCCC(C1)N2C c1(C(N(CC)CC2CCCCN2C(=O)COC)=O)cccc(Cl)c1[N+](=O)[O-] N1(Cc2c(C)n(C)nc2)CCC(F)(c2cccc(C(F)(F)F)c2)CC1 CN1CCCc2cc(CNC3(CC(F)F)CCNC3)ccc21 N1(C(CN(C(=O)OC)C)=O)CCC(CCNC(=O)C(O)c2cnc[nH]2)C1 CCC1(C(=O)N2CCOC(C)CC2)CCCc2ccccc21.N(C)C C12(C(N3C(CCN(C(c4cnc(C)nc4)=O)C)CCCC3)=O)CCC(F)C1CC2 N1(C2N(C(=O)NC3C4COCC34)CCCC2)Cc2ccccc2C1 N1(C(c2nc(C)oc2)=O)CC2(COC(CNC(c3cc4c(nn3)CCC4)=O)C2)C1 c1(CN(C)CC2CCS(=O)(=O)C2)ccnc(C2CCN(C(=O)OC(C)(C)C)C2)c1 c1(OC)ccc(C(=O)NCC2C(C)CCN2C(C2CN(S(N)(=O)=O)C2)=O)c(Cl)c1 C12(C(=O)NCCN(C(C(C3CC3)OC)=O)C)CCC(CO1)C2 C1(NC(c2c(C)nn(C)c2C)=O)CC2CC(C1)N(C(c1cocc1C(N)=O)=O)C2 N1(C(C2(NC(C3(C)CC3C)=O)CC2)=O)CC(COC(C)C)CC2OCCC12 N1(C(CCC=CC(C)C)=O)C2CCC1CC(F)(CNC(c1ccncn1)=O)C2 CCC(O)C(C)(C)C(=O)NCCCN(C)C(c1ccoc1C1CC1)=O c1(C(C)C)ccc(CNC(C23CC2CN(Cc2cnc(Br)o2)C3)=O)cc1 C1(C(N(CCN(C(C)C)C(C2CC(S(C)(=O)=O)C2)=O)C)=O)CC(=O)OC1(C)C n1(CC(=O)NC2(C)CCN(C(c3cnn(C)n3)=O)C2)ccc(=O)c([N+](=O)[O-])c1 C1(CNC(c2cnn(C)c2)CCOC)CC(=O)C12CCC2 Cc1cccc(-c2nc(C)c(C(=O)NCC3CC(NC(=O)C(N)=O)C3)[nH]2)c1 N1(C(CC(=O)NCC)=O)CC2CC(NC(c3nc(C)ccc3OC)=O)C2C1 C1(C(N2C(C)(CNC(C(C(=C)C)(C)C)=O)CCC2)=O)CCC(=O)CC1(C)C N1(C(C(=O)NCCOC)=O)CCC(O)C(C(=O)NCC(C)CC(=O)OC)C1 N1(C(CC(C)C2CCCC2)=O)CCCC12CCCN(C(C1CCCO1)=O)C2 CC1CCCC(C(=O)NCc2cc(C(=O)NCc3cn(C4CC4)cn3)n[nH]2)C1 C=C=CC(C)C(=O)NCC=CCC1(CNC(=O)CCc2csc(Br)c2)CC1 C1(C)(C(=O)NCC2CN(c3nnc(C(=O)OCC)s3)C2)CCc2ccccc2C1 C1(C)(NC(CN(C(COC)=O)C)=O)CC(NC(=O)C(C)Cn2ccnc2)C1 C(CCF)(C(=O)NCCc1nc(C)cs1)NC(C(C)SCC)=O CCCCC(O)CC(=O)NCC1CCCN(C(c2ccc([N+](=O)[O-])o2)=O)C1 c12ccccc1C(C)N(C)C(=O)OC2.C1(C(=O)O)(CO)CCOC1CC.C(C)(C)(C)SCBr.C CC1=NOC(C)(CNC(=O)C(c2ccccc2Br)(F)F)C1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(CCC)N(C(=O)CC(=O)NCC2CC2)CC1 CC(CS(C)(=O)=O)C(=O)N1CC(C)(C)CC1CNC(c1ccnn1C)=O C(=O)(CCCS(C)(=O)=O)NC1(C(=O)OC)CCCN(C(=O)C(C)O)C1 N1(C(COCC)=O)CC(NC(=O)CNC(C2CCCC2)=O)C2CC2C1 CC(C)C(C(=O)N1CCC(O)(CN(C)C(c2coc(Cl)n2)=O)C1)NC(N)=O C(C(C)(Cn1cccn1)NC(=O)CNS(N)(=O)=O)NC(C(OC)OC)=O NC(CCF)C(=O)NCc1ccc(-c2cccc(C(F)(F)F)c2)o1 CC(Cc1ccccc1)CC(=O)NCC(C)(C)CC1CN(C(c2ccn(C)n2)=O)C1 C(=O)(CCCCCF)N1C(CCNC(C=Cc2ccc(C)o2)=O)CCC1 CN1CCCCC1CC(=O)NCC1CCC1NC(c1cc(Cl)sc1Cl)=O CC(CCC(=O)N(C1(CO)CCOCC1)C)NC(=O)CSC1CC1 c1(C(C(=O)NCCOCC)N(CC(C)OC)C)ccc(N(C)C)nc1 C(C1=Nc2ccccc2S(=O)(=O)N1)NC(=O)NC1CCC1c1c(Cl)cccc1Cl CC1CC(CNC(c2c(F)ccc(Br)c2Cl)=O)CC(F)(F)C1 C1(C(=O)NCC2C(C)CCCN2C(C2OCC2(C)C)=O)CCc2n[nH]cc2C1 c1(C(=O)NCCOCCNC(C2COC(CC3CC3)C2)=O)ccncc1Cl c1(C(CNC(C2CC2(F)Cl)=O)=O)ccc(F)cc1 C1(NC(c2nn[nH]c2C(F)(F)F)=O)CN(C(c2ccc(CO)nc2)=O)CC1O N1(C(CSS(C)(=O)=O)=O)CCCN(C(c2ccnn2-c2ccccc2)=O)CC1 CS(=O)(=O)CCC(=O)NC12CC(NCc3cncc(C#N)c3)(C1)C2 N1(C(c2cn(C)nc2)=O)CCC2(NC(c3cncc(F)c3Cl)=O)CCCCC12 CC1(C)CC(=O)NCC1C(N1CCC(CF)(NC(=O)C(N)=O)C1)=O Cc1cc(C)c(C(N2CC(C)(NC(=O)C(C)ONC(=O)OC(C)(C)C)C2)=O)s1 c1(CC(=O)NCCCC(C)NC(CNC(=O)OC)=O)ccncc1Cl Cc1cccn2ncc(C(N3CCC(C)(CNC(c4cnc(Cl)s4)=O)C3)=O)c12 N1(C(C2CC(C)CC(C)C2)=O)CC2CC(NC(c3cnn(C(C)C)n3)=O)CC1C2 CC(C)(C(=O)NCC1CCN1C(c1cccc[n+]1[O-])=O)S(C)(=O)=O C(N=c1ccc2nnnn2[nH]1)C1C(NC(=O)OC(C)(C)C)N(C)C(=O)C1 c1(OCC)cccnc1C(=O)NC1CCC(F)(CNC(=O)C(F)n2ccnc2)C1 c1(NC(C)=O)cc(N2CCSCC2)nc(S(C)(=O)=O)n1 CCCC(C)CC(=O)NC(c1ccccc1)CNC(=O)C#CC1CC1 c1(C(C(=O)NC(C2CN(C(c3ccn(C4CC4(F)F)n3)=O)C2)C)O)cnn(C)c1 N1(CC)CCCC2(CCN2C(=O)C(c2cccc(F)c2Cl)(F)F)C1 N1(C(C)C)CC(NC(c2c(CN)nnn2C)=O)C(C)C1.C(C)(C)(C)OC=O CC1CC(CNC(=O)Cn2cc(C3CC3)cn2)CN1C(C1CC(C2CC2)C1)=O C1(NC(=O)CCSC(F)(F)F)CC2(CCN(C(=O)Cc3nncs3)CC2)C1 C12(CNC3C(OC(CCC=CC)=O)COC3)CC(C(=O)OC)(C1)C(C)O2 N1(C(CC=C)=O)CC(F)CC1CN(C)C(C1(C(F)(F)F)CCCCO1)=O C1(OC)CC(CNC(=O)C=CC(C)SC)N(C(=O)C=CC2CCOC2)C1.C(C)(C)(C)O c1(OC)cccnc1C(=O)NCC(C1CCC1)NC(C1CC1c1ccc(C)s1)=O C1(NC(C(CC)OCC)=O)CCN(C(c2cnc(CC)nc2O)=O)CC(C)(C)C1 n1(CC)nc(C(=O)NCC2CN(C(=O)CCc3cn(C)cn3)C3CC23)cc1O N(C(=NCC1(CSC)CCCC1)N1CCC2=C(CCCC2)C1)C(COC)C N1(C(CCc2n(C)ccn2)=O)CCC2(CCN(C(c3cc(Br)cn3C)=O)C2)C1 Cc1cc(C(=O)NCC2(C)CC(F)(F)CN2C(=O)CCF)c2c(C)nn(C)c2n1 c1(C(=O)N(c2ncc(I)cn2)CC2CCCC2)cnc(C2CC2)nc1 N1(C(c2n(CC)ccn2)=O)CCC2CCN(C(=O)C(C)C#N)CC2C1 N1(C(CCCC=C)=O)CC(C)CN(C(c2cc(C(F)(F)F)c[nH]2)=O)C(C)C1 c1(NC(C(CC)NC(N)=O)=O)nc2c(s1)C(C(C)C)OCC2 C(CCCN=c1nc(O)c(Br)c[nH]1)NC(C(C(C)C)NC(N)=O)=O C(=O)(C(C(C)(C)C)N(C)C)N1C(C(=O)N(C2CCC3CC23)C)(CC)CCC1 Cc1cccc(C(c2ccccn2)NC(c2snnc2C2CCC2)=O)c1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(C3CC=CCC3)=O)CC21 c1(C(=O)NCCC2CCCCN2C(c2nnc(O)s2)=O)ccc(F)c(F)c1 C1(N(C(=O)C=C2CC2)CC)CC2CCC(C1)N2C(C1(NC(N)=O)CC1)=O C(C(F)(F)C(F)(F)F)C1CN(CCc2cn(CS(CCc3ccc(C)cc3)=O)nc2)C1 c1(C(=O)NC2C=CCN(C(c3c(C)cc(SC)o3)=O)C2)cnc2cccnc2c1 CN1CCCC1(C)C(=O)NC1CCOCC1C(=O)NCC12CCC(CO1)C2 C(CC(F)F)(C(=O)NCCC1CCCC1)NC(c1csc(O)n1)=O N1(C(c2cnc(C)[nH]2)=O)CCC(N(C(=O)CN2CCCNC2=O)C)CC1 C1(NC(C2N(C)CSC2)=O)CCN(C(c2cc(O)ncn2)=O)C12CC2 N1(C(c2cncc(OCC)c2)=O)CCC2CCC(NC(=O)C=C(C)C)C1C2 C(=O)(C(C)(COC)CC)NC(CCCC)CNC(c1cncc(CO)c1)=O N1(C(c2cccc3occc23)C(=O)Nc2c(C)c(Cl)ccc2)CCCCC(C)CC1 c1(OC)cc(F)c(C(N2CC(NC(c3nccnc3N)=O)CC(F)C2)=O)cc1N c1(C(N2C(CNC(CSCC(=O)OC)=O)CC(OC)C2)=O)cc2n(n1)CCCO2 n1(CC)ncc(C(=O)NC2(C(=O)NC(c3cn(C)cn3)C)CSC2)n1 c1(C(N2C(C)CC(CNC(CN(C(C(C)C)=O)C)=O)C2)=O)ccc2c(c1)NC(=O)C2 C(=O)(CCCC(F)(F)F)N(CCC(C)NC(c1c(SC)n(C)nc1)=O)C CCCCC(O)CC(=O)N1CC2CCC1C(CNC(C1(C(N)=O)CC1)=O)C2 CC1CC=C(C(=O)NC23CCCN(c4ncc(Br)cn4)CC2C3)CC1 N1(C(C(CC=C)C)=O)CCC(F)(F)C(CNC(=O)CCCC2CCOCC2)C1 c12cnc(C#N)c(c1)C(=O)N2.Cc1ccc(C(=O)Nc2cccc(CO)c2)nc1 Cc1nn(C)c(Cl)c1C(c1nnnn1CC1CCOC1)NCC1CC1 c1(N(c2ccc(C(F)(F)F)cn2)Cc2cccc(O)c2)ncnc2c(Br)csc12 O(NC(=O)C(C)(C)C1CN(C(c2cccc(CO)c2C)=O)C1)CC CC1COCC(C(N2CC(C(=O)NCCC(C)c3cn[nH]c3)C(C)C2)=O)O1 Cc1ccnn1CC(=O)NC(CNC(=O)CCc1cn[nH]c1)C1CC1 C(Cn1ccnc1)CN=c1ccnc(NCCCc2cccnc2)[nH]1 C1(NC(CC(c2cccc(F)c2)C)=O)CCCCC1NC(C1(C(=O)N(C)C)CC1)=O CS(=O)(=O)c1cccc(C(CO)NC(c2cc(O)cc(O)n2)=O)c1 c1(C(=O)NC2CC(C)(NC(C(CC)C#N)=O)C2)cc(Br)cc2nc[nH]c12 c1(C(N2C(CN(C(=O)C3=CCCC3(C)C)C)CCC2)=O)cnn2c1C(=O)NCC2 C(c1cnccc1C)=CC(=O)NC1CC(CNC(CC2C(C)=NOC2=O)=O)C1 FC1(F)CC(CNCc2cc3nncn3cn2)CC(c2ccccc2)C1 n1(CCC(=O)NCC2CC(CNC(C3(CCO)CC3)=O)CO2)cccnc1=O c1(OC)cc(C(N2CCC(CF)(NC(=O)C=CS(C)=O)C2)=O)cnc1O C1(C(=O)NCc2cccc(CN3CCCCC3)c2)CCCN(CC(F)(F)F)C1=O Cc1ccc2c(n1)N(C(c1c[n+]([O-])ccc1[N+](=O)[O-])=O)CCO2 C12(c3nc(COCC)nn3C3CCS(=O)(=O)C3=O)CCCC1C2(F)F N1(C(=O)C(O)C2CCC2)CCCC(N(CCO)C(C2(Cl)CC2(F)F)=O)C1 CC1(C)CCCC(CNC(N2CCN(C(c3ccc(F)cn3)CN(C)C)CC2)=O)C1 c1(NC(=O)OC(C)(C)C)cc(C(F)F)cc(F)c1.c12ccc(cc1)COC(=O)C2 Cc1noc(C)c1S(=O)(=O)NC(c1cc(CN)on1)=O CC1CN(C(c2csc(=N)[nH]2)=O)CCC1NC(=O)CC1CC(C2CC2)C1 Cc1nc(CN2CCC(NC(c3cnc(C)n3C)=O)C2)n(C)n1 CN1CCC(C(=O)NC2(C)CCCN(C(c3cccnc3N(C)C)=O)C2)CC1=O C12(C(=O)NCC3CCN(C(C4(CN(C)C)CC4)=O)C3)CCCCC1C2Br C1(CNC(Cc2nc(CCOC)sc2)=O)CC(OC)CN1C(=O)CC1CC1 N1(C(c2ccn(CC)n2)=O)CCC(C)C1C(=O)NOCC=CCl C(=O)(C(C(C)C1CC1)N1CCC(CN(C)C)CC1)NCC C(C(C)(C)C(=O)NCCCC(C)O)N(C(c1c(C)scn1)=O)C C1(C2CCN(C(=O)CN(C(=O)C(C)C)C)C2)(NC(C(C)OCC=C)=O)CC1 c1(C(=O)NC(COC)C(=O)NC(C)Cc2nccn2C)ccn2ccccc12 CCCC(C)(O)CC(=O)N1CCC(C)(C)C1C(=O)N(C(C)CC(=O)OC)C C(=O)(C(C)(C)CC(=O)NC1CN(C(=O)C(C)C2CCCC2)CC12CC2)OC C1(C)(NC(C(COC)(C)OC)=O)CCN(C(c2ncc(C(N)=O)cc2Cl)=O)CC1 c1(C(C)C)ccc(C(C)CC(=O)NC2CCCC2Oc2ccccc2)cc1 c1(C(=O)NCCC2CCCCN2C(C2CCCO2)=O)ccn2c1CCC2 c1(C(=O)NCC2(NC(c3cnsn3)=O)CC2)cc(Br)ccn1 CCCCCC(C)CC(=O)NC(C)CC(C)NC(C1CCN(C)CC1)=O c1(CNC(c2cnc(O)[nH]2)C)ccc(F)nc1 C1(NC(c2coc(C(F)F)n2)=O)(CNC(c2ccsc2C(F)(F)F)=O)CCOC1 C1(CC(=O)N(C(C)C(C)(C)O)C)CN(C(c2coc(CO)c2)=O)CC12CC2 CCC(CC(=O)NCC#CC(=O)NC1CC12CCCC2)C1CC1 CC1CC(CNC(=O)CCCN2CCCC2)CN1C(c1cc(C#N)c[nH]1)=O CS(=O)(=O)CC(=O)NCC(O)CCNC(=O)CC(=O)NCC(F)(F)F.C(=O)C=CC#N c1(CCC(=O)NC2CC(C(=O)NCC3CCNC3=O)C2)ccc(C(F)(F)F)cc1 N1(C(C(=O)Nc2cncc(OC)c2)=O)CC2CC(OC)CC2C1 CCCCCC(O)C(=O)NC(C(=O)N1CC(F)C1)C(C)(C)O C1(S(C)(=O)=O)(C(=O)NCC2CN(C(C3N(CC)CC3)=O)C2)CCCC1 C1(CN(C)CC2CCCN(C)C2c2ccnn2C)CCC2CC1C2(C)C N1(C(N2CCC(OC(F)(F)F)CC2)=O)CC(C2CC2)C(F)(CO)C1 C=C(Cl)C(C)(C)C(=O)N1CCC(CCNC(=O)Cc2n[nH]c(=N)s2)CC1 C12CCC1NC(=O)N2.C(C(C)N(C)C)N(CC)CC C(C)(CCC(=O)N1CC(OC2CCN(C(=O)C(Cl)=CCl)CC2)C1)SC c1(OC)cc(C(=O)NC2CCN(Cc3csc(Br)c3)CC2F)ccc1CO CC(C)CCC(C)NC(=O)CC1CC1CNC(C1CC2(CSC2)C1)=O C(=O)(C(CCC(C)C)NC(=O)CCCC(=O)N(C)C)NCC(COC)C(C)C C(CCCCCC(=O)N1CCC=C(F)C1)NC(CCCCCN(C)C)=O N1(C(c2c(Cl)ccc(OC)c2)=O)CCCC(N=c2ccnc(C(F)(F)F)[nH]2)C1 C(CCC(C)C(=O)NC1CCN(C2CCCCC2)CC1)OC.c12nnc(o1)CO2 C=C1c2ccccc2C(=O)N1CC(N1CCCCC(NC(c2ccco2)=O)C1)=O c1(C(=O)NCC(C)CNC(C2CC(=C3CCC3)C2)=O)ccnn1CC(F)F C1(C(=O)NCC(C)(C)N(C)C)CCCCN(C(C2CCC3CC2CO3)=O)C1 c1(NC)ccc(C(N2CC3C(C(=O)NCCc4csnn4)C3C2)=O)cc1 N1(C(c2c(C)snn2)=O)CCN(C)C(C(=O)Nc2cnc(F)nc2)C1 CC1(C)CC(C(N2CCCC2CCCNC(c2ccncc2)=O)=O)CC(C)(C)O1 N1(c2ncc(C(=O)OC)nc2)CCC(CNC(c2cccc(F)n2)=O)C1(C)C N1(CC(=O)NCC(C)(C)OC)CCN(C(=O)C(F)n2ccnc2)CC1 C1(NC(C2N(C(c3c(CC)cc[nH]3)=O)C(C(C)C)CC2)=O)CC2CC1C(O)C2O Cc1cc(O)c(CN2CCCC(N(C)C)C2)cc1Cl.c12nc(Cl)ccc1C(=O)N2 C#Cc1cccc(CCC(=O)NC2CN(c3ncncc3C#N)C2)c1 C1(C(=O)NC2CC2NC(=O)CCCc2ccc(O)cc2)(CC)CCNC1=O CC1CN(C(c2cc3ccccn3n2)=O)CC(C)C1NC(=O)CC=CC(C)(C)C C1(NC(c2ccc(CSCC)cc2)=O)CCC2CN(C(C3CC3F)=O)CC2C1 N1(C(CSC)=O)CC2CCC(NC(C3CCCSC3)=O)CC2C1 c1(C(=O)NCC(CC=C)NC(=O)C(O)CSC)nccc2ncncc12 c1(C(N2CC(CNC(COC3(C)CCC3)=O)C2)=O)cccc(C#N)n1 c1(OC)cccc(Cl)c1C(=O)NCC(C1CC1)NC(c1cc2n(n1)CCC2)=O N1(C(=O)Nc2ccc(CO)cc2)CC2CN(C(c3ccc(Cl)cn3)=O)C2C1 C12(CNC(=O)CN3CCCC3=O)CCCC1CN(C(C1CCCO1)=O)C2 c1(C2(NC(=O)NCC3(O)CCOC3)CCC2)ccccc1F C1(NC(=O)CCN2CCOCC2)CC2CC1CN2C(=O)Cc1cnoc1 N1(C(C2CNCCN2Cc2cccc(Br)c2F)=O)CCCC2(CCOC2)C1 C(CC(=O)N1CCCC(C)(C)C1)(C(F)F)NC(C(C1CC1)OCC)=O C1(CC=C)(C(=O)N(C2CCN(C)C2=O)C)CCN(C(=O)Cc2ccccc2F)C1 C(=O)(CCC(=O)NCC(O)CNC(C1CC=CCC1)=O)Nc1nnc(C(C)C)s1 c1(CCC(=O)NCC(CC)NC(c2coc(C)c2)=O)cccnc1C C(=O)(CC(O)CC(C)(C)C)N(CCC(=O)N(CC(=O)OC)CC(C)C)CC=C c1(C(=O)NCC(CC=C)NC(C2CC(C(C)(C)C)=NO2)=O)ccc(F)c(F)c1F CCC(CC(=O)NC1CCCC(C(=O)NCC(C)(C)OCCOC)C1)OC C(=O)(C(O)CC(N)=O)N1C(C(=O)NC(C#CCC)(C)C)C=CC1 CC1(C)C(CO)CCN1C(=O)CCC1CCOC1.N12CC(C)(C1)NC2=O c1(C(=O)NCC(CNC(C(C)(C)NC(=O)OC)=O)O)cc2nnn(C)c2s1 c1(C(=O)NC2CCC(NC(CC3CC(=O)C3)=O)C2)cccc(-c2ccccc2)n1 C=C(Cl)CC(C(=O)Nc1cnn(CC)c1)NC(=O)CCC(N)=O c1(C(=O)NCC(CNC(c2ccc(N(C)C)cc2)=O)(C)O)cc2occc2[nH]1 C1(C(N(CCOCC=C)C)=O)COC2(C1)CN(C(=O)C(F)C(CC)CC)C2 N1(C(=O)Nc2ccnc(OC)c2C)CCc2c(ccnc2O)C1 C1(CCC=C)(C(=O)NC2COCC2CCO)CN(C(c2ccoc2CC)=O)C1 c1(C(=O)NC(C2(CC)CC2)C)[nH]nc(C(=O)NCC2CC2c2ccn(C)n2)c1C Cc1c(C(N2CC(C(N)=O)(CNC(C3CCCOCC3)=O)C2)=O)cccc1O c1(C(=O)NC2CCC(NC(C(COC)NC(C)=O)=O)CC2)ccnc2[nH]cnc12 N1(C(=O)NC(c2cccc(Cl)c2F)C)CCC(F)(C(F)F)CC1 N1(C(CCN(C(C2CC3CCC2O3)=O)CC)=O)CCC2CC1C(=O)O2 c1(CNC(c2c(NC(=O)Cc3ccco3)cnc(Cl)c2)=O)cccc([N+](=O)[O-])c1 C1(C)(C(=O)OC)CC(C(=O)NCC(O)CNC(C2(C)CCC2)=O)C1 c1(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccc2nsnc2c1 C(=O)(C(CCC(N)=O)N(C)C)N1CC(CCNC(c2c(C)occ2)=O)C1 c1(C(N2CC(COCC(=C)C)C2)C)cccc(C)c1.C1C(=O)O1 C(C1=CCN(C(C2CC(OC)(OC)C2)=O)CC1)NC(C(C)NC(CC)=O)=O N1(C(CC(=O)N(C)C)=O)CC2CC2(C(=O)NCCc2cc[nH]n2)C1 C(C(=O)NCC1(O)CCC(C)C1)(C(C)(C)C)NC(CC1CCC(C)CC1)=O CCC(CCCC(=O)NC1CC(=O)NC1=O)NC(=O)C(C1CCCCC1)C C12OCCN(C1C)C2.C1(OC)CCC(=O)CC1 Cc1c(C(=O)NC2CC(C(C)NC(=O)CCc3ccccc3F)C2)[nH]ccc1=O Cc1conc1C(N1CC(CNC(c2cccn2C2CCCC2)=O)C1)=O N1(C(=O)CC2CCCCCC2)CCC2(C(N3CCC(F)(CF)C3)=O)CCCC12 c1(C(=O)NCC2CCCN2C(C2CCCCO2)=O)nc2c(s1)COCC2 N1(C(C(C(CC)O)C)=O)CC2(CCN(C(C3CCCC3C(F)(F)F)=O)CC2)CC1 C1(C(N2CC(C(N)=O)(CNC(c3cc(CCO)on3)=O)C2)=O)CCCC(O)C1 C1(NC(C2(C)CC(=C)C2)=O)CN(C(c2cccc(OC(C)C)c2)=O)C2CC12 CC1CN(C(c2cn(C3CC3)cn2)C(=O)NCCC#N)C(C)(C)C1 Cc1oc2nc1C(=O)N1CC2C1.C1(CNC(=O)OC(C)(C)C)CCC(C(C)C)CC1 c1(C(=O)NCC(CC(C)C)NC(C(C(C)C)SC)=O)ncc(Br)cc1O c1(C(N2C(C(=O)NCC(=O)N(C)C)C=CC2)=O)nc(Br)ccc1F N1(C(C2CCC(C)CC2)=O)CC2CC3CC2C1C3NC(c1cc(F)n[nH]1)=O C(=O)(C(=O)C1CC1)NCCC1(CNC(=O)OC(C)C)CC1 c1(C(=O)NCC2CCC(C(=O)NC3CC3)CC2)ccnc(NC2CCCC2)c1 C1(NC(CCC2C(C)(C)C2)=O)CC2CN(C(c3ccc4sncc4c3)=O)CC2C1 C(=O)(C1CCCn2nccc21)NCCN(C(C1(C(C)(F)F)CCC1)=O)C1CC1 C=C(Cl)C(C)(C)C(=O)NC1CN(C(=O)CCCCCc2ccc(F)cc2)C1 c1(C(=O)NCC(C)NC(=O)C=C(C2CC2)C2CC2)cnc(O)c(C(F)(F)F)c1 c1(C(=O)NCCN(C(=O)C(C2CCCCCC2)F)CCC)c(C)cc(C)nc1S c1(C(=O)NCCC(CSC)OC)nn(C)c(=O)cc1C.c12csc(c1)C(=O)NC2 c1(N2CCCC(C)(CSC)C2)nc(=NCC2CCC(C)N2C)[nH]c2cc[nH]c12 C=C1CCN(C(=O)C2=NOCC2)C(C(=O)NC2CCNC(=O)C2)C1 c1(C(N2CCC(NC(C(CC)CC(C)C)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1N S(=O)(=O)(c1cccs1)NCCC(=O)N(C(CNC(C(C=C)(C)O)=O)C)C C1(C(=O)NC2CC(OCC)C2)CC12CCN(C(C1(F)CCCCC1)=O)C2 C1(N(C)C(c2cncnc2)=O)Cc2ccccc2N(C(C2C(C)(C)C2(C)C)=O)C1 C1(CC(=O)NCC2CC(NC(Cc3n(C)ccn3)=O)CC2O)CCOCC1(C)C c1(C(CNC(C2CCNC2=O)=O)NC(c2ccnn2CCF)=O)ccc(F)cc1 c12ccc(nc1)NS(=O)(=O)C2.c1(-c2ccc(C)o2)ncc(-c2ccccc2)s1 c1(OC)nccc(C(N2CCC(NC(c3cc(N)cnc3Cl)=O)C2)=O)c1Br N1(C(C(C2SC(=N)NC2=O)C)=O)C2CCC1C(C(=O)NCCCOC(=N)O)C2 C(CCN=C(NCc1ccc(-n2cccn2)nc1)NC(c1ccco1)C)SC C1(NC(c2ccc(C)s2)=O)CC2CC(NC(=O)C(F)OC(F)(F)F)C1C2 c1(C(N2CC(C)(NC(c3cc(CO)on3)=O)C2)=O)ccc(-c2nnco2)cc1 C1(CC)CN(C(C23CCC(C2)C3)=O)CC1C(=O)NC1CCCN(C2CC2)C1 Cc1ccc(F)c(C(=O)NCC2(F)CCC(CNC(=O)C(C)C3CCC3)CC2)c1 C1(C(=O)NCCNC(c2cc(C)nn2C(F)F)=O)COc2cc(F)ccc2C1 c1(C(N2CCC(c3ccc(C#N)s3)C2)=O)cccc2c1CNCC2 c1(C(N2CC(CNC(C3C(C)C3)=O)C(C)(C)C2)=O)cncc2cc(Cl)ccc12 C(N=c1[nH]c(=NCCC#CCO)[nH]c2c1COC2)C1(OCC)CCCC1 c1ccc2c(c1)CCN(c1ccnc(NCc3cnc(C4CC4)o3)n1)C2 C1(CC)CN(C(=O)C(c2ccc(Cl)cc2)C)CCN1C(C1CC(=C2CCC2)C1)=O CC1(C)CN(C(C2CCC23CCC3)=O)CCC1NC(c1n[nH]cc1Br)=O c1(CNC(CCC)=O)ccc2c(c1)CCCC2NC(C1CCC12CCCO2)=O N1(C(c2cnc(OCC)c(Cl)c2)=O)CCC2CCCN(C(=O)COC(F)F)C2C1 C(=O)(C1CCCc2scnc21)N1CC2=C(CN(C(CSCC(=O)OC)=O)C2)C1 N1(C(=O)OC(C)(C)C)CC(CNC(C2(n3nccn3)CC2)=O)CC1(C)C N1(C(c2c(C)sc(C(F)(F)F)n2)=O)CCC(NC(C23CC(C2)C3)=O)C(CO)CC1 C1(NC(C(=O)NC(CC)CNC(=O)C(CC)n2ccnc2)=O)CCN(C)C(=O)C1 N1(C(C)=O)CCC(NC(c2nc(C)oc2N(C)C)=O)CC1 CC(N=c1cc[nH]cc1S(=O)(=O)NCCS(=O)C(C)(C)C)CC(C)(C)C CC1(C)C(NCc2ncc(-c3ccccc3)s2)CC1Nc1ncccn1 N1(C(CC(CC(C)C)C)=O)CCN(CCNC(C2CC(C)(C)C2)=O)C2(CCC2)C1 N1(C(C2(COC)CC2(F)F)=O)CCC(O)(C(F)(F)CO)CC1 N1(C(CCC#CC)=O)CCCC12CCCN(C(C1CCCN1CC(F)(F)F)=O)C2 CC1(C)CCCC(O)(C(=O)NC2CCCN(C(=O)C(F)=CC3CC3)C2)C1 CC1CCC(NC(c2cc(O)nc(Cl)c2)=O)CN1C(c1ccc(C(F)F)cc1)=O C1(C(=O)NCCC(C)(C)NC(C(CC)SC)=O)Cc2ccc(F)cc2O1 C(C(=O)N1CCCC1)(C(C)C)NC(CCCNC(C)=O)=O.C1(CO)CCCS1(=O)=O C(=O)(C(C(C)(C)CC)OC)NCC(CC)NC(=O)Cc1cnccc1C CC1CN(C(=O)C(C2CCCO2)C2CC2)CCN1C(=O)C=CC1CCOC1 N1(C(=O)COCc2ccc(F)cc2)CCN(C(=O)C2=COCCO2)C2(CCC2)C1 C=CCC(CNC(c1ccc(F)c(I)c1)=O)C(=O)N1CCCCC1C N1(C(C(C)C)=O)CCCCC1C(=O)NCC(C)NC(c1csc(C(=O)OC)n1)=O c1ccc(CCNCc2ccc(Cn3ccnc3)s2)cc1 N1(C(CCCC=C)=O)CC(NC(=O)CC2CSCCO2)C2(CCS(=O)(=O)CC2)C1 C(C(C)(C(=O)NCCc1cccc(O)c1)NC(c1cnc(S)nc1)=O)SC C1(C(N2CC(O)(CNC(C3(C4CCCCO4)CCC3)=O)C2)=O)CCCCC1F CCC(C)(C(=O)NCC1CN(C)CCN1C(=O)CC1(NC(=O)OC)CC1)C(F)F C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C)C(CNC(=O)CSC(C)(C)C)C1 c1(C(=O)NC(C2CCN(C(c3cc(C)c(C)s3)=O)CC2)C)cccc2ccnn12 C1(CC)CN(C(=O)CC#N)CCC1C(F)(F)F.c12cnc(nc1)CNC2=O c1(C(=O)NCC(C)CNC(C2(C(F)(F)F)CC(F)(F)C2)=O)cc(F)cc(F)c1 C1(C(N2CCC(C)(NC(C(c3ccc(C)cc3)=O)=O)C2)=O)CC12CCSCC2 N1(C(C=C(C)C2CC2)=O)CCC(O)(C(C)NC(=O)Cn2cnc([N+](=O)[O-])n2)CC1 C(C(CC(=O)NCc1ccc(F)cc1)OC)N(C(C1(C(=O)OC)CC1)=O)C Cc1ccc(C(=O)NCC2CC2CNC(=O)COc2ccc(F)cc2F)c(=O)n1C c1(C(=O)NCC(O)CC2CCCO2)ccc2nnc(-c3ccccc3)n2c1 C12(NC(C(C)C#N)=O)COC(C(=O)NCCC(=O)NCc3ccc(F)cc3)(C1)C2 C(CNC(C1CCCN1Cc1cccc(OCCCl)c1)=O)(C(C)(C)C)NC(C)=O C(CC(C)CC)(C(=O)NCc1nccc(C)c1F)NC(c1c(CC)nc(C)o1)=O C1(NC(C2CC(OCC)C2)=O)CC2CC(NC(=O)C(CC)NC(N)=O)CC12 c1(C(=O)NC(CNC(CSCC)=O)(C)CC)cncc(O)c1 C(=O)(CCCCCCCC1CC1)N1CCC(N(C(c2ccoc2Br)=O)CC)C1 C(C(CN=c1[nH]n(C)cc1[N+](=O)[O-])C(F)(F)F)NC(C1CCN(C(C)C)CC1)=O CCC(CN=c1nc(N2CCC(C)(CC)C2)c2ccc(OC)cc2[nH]1)C(C)C c1(N(C)CCO)ccc(S(=O)(=O)NC2CC2)cc1Br.C1(N)CCC1C(C)(C)C C(=O)(CC(C(F)F)NC(=O)CC1CC(F)(F)C1)NCC(C)OCCO N1(C(c2ccn(C)c2)=O)CCOCC2(C1)CN(C(=O)C1CC1)CCCO2 c1(OC(C)C)ccc(C(=O)CN2CCC(CN3CCC3)C2)cc1Cl C1(C(=O)Nc2nnc(C(=O)OC)s2)CCN(C(c2cc(Cl)ccc2F)=O)CC1O c1(C(N2CC(N(C(=O)C=CCn3cncn3)C)C(F)C2)=O)cc2scnc2[nH]1 C1(CNC(CNC(C(C)(C)C)=O)=O)CN(C(=O)CCNC(N)=O)C2(CCC2)C1 Cc1csc(C(C)C(N2CC=CC2CNC(=O)CCCC2CCC2)=O)n1 c1(CC(N2C(CNC(CCC)=O)CCCCC2)=O)cc(F)c(OC)c(S(N)(=O)=O)c1 C1(CCC(=O)NC2CCCC2CNC(C2(O)CC2)=O)CCC(=O)N1 CCC(CC1CCCCC1)C(=O)NCCN(C(=O)C(c1cccc(Cl)c1)OC)C c1(C(N2CC(NC(CC3C(C)(C)CC3)=O)C2)=O)cc(O)ccc1Br N1(C(CCC2C(C)C2)=O)CCC=C(C(=O)NCCC(Cl)Cl)C1 c1(C(=O)NC2CCC(N(C)C(C3CCCC34CC4)=O)CC2)cc2n(n1)CC(F)C2 N1(C(CC2CCC(=O)N2)=O)CC(C2CCCN(C(=O)C(F)(F)c3cscn3)C2)C1 c1(C(=O)NCC2CN(C(c3cc(OC)c(F)cc3)=O)C2)cnc2c(c1)CCCO2 C1(C(=O)NCCCC(F)(F)CO)CC12CCN(C(c1ccccc1)=O)C2 c1(NC(C)=O)ccc(C(=O)NC2CC2NC(C2CC(O)C2)=O)nc1 C1(CC(=O)NCC(C)C2CCC2)CC(O)CN1C(=O)CN(C)C1CC1 c1(C(=O)NCCC2CCCN(C(C3(C)COC3)=O)C2)ccc2cc(F)ccc2n1 O=S1(=O)CCN(Cc2csc(-c3ccccc3)n2)C(c2cccs2)C1 C(=O)(CC(C)(C)C(C)(F)F)N1CCC(NC(c2c(CC)cccn2)=O)C(C)C1 c1(CC)cc(NC(C2(NC(C3(C)C=CCC3)=O)CC2C)=O)cnc1C C(=O)(C(CC)(CO)OC)N1CC(C(C)(CCC(=O)OC)NS(CCCC)(=O)=O)C1 CC(CC(=O)NCCCN(C1CCCC1)C(c1cc2scnc2[nH]1)=O)C(F)F C1(CNC(C2CCOC2)=O)CCCCN1C(=O)C=C1CC1 Cn1cc2cccc(-c3nc(C4CCCO4)nn3Cc3ccccc3)c2n1 n1(CC)cc(CC(=O)NCC2C3CN(C(C4(C)CCC4)=O)CC23)c(C)n1 c1(C(=O)NC2(CCNC(c3c(C)cc(N)s3)=O)CCC2)cc2c(=O)[nH]ccn2n1 C(=O)(CCCC(=O)NC1CC(O)(CNC(=O)C=Cc2ccco2)C1)N(CC)CC Cc1cnn2cc(C(=O)NCC3CN(C(C4COCCO4)=O)CC3O)cnc12 CN1CCC(C(=O)NCCCOCCCNC(=O)C#CC2CC2)C1=O c1(C(=O)NC2CCN(C(C3(CCC=C)CC3)=O)C2)cc(C)cnc1N CCC(CC)(CC)C(=O)N1CC2CCC1C2NC(=O)C(C)SC c1(NC(C(=O)NC2CC(C(=O)OCC)C2(C)C)=O)ccc(Br)c(C)c1 c1(C(N2CC(C)(C)C(NC(=O)C(O)CF)CC2)=O)cc2c(cc1N)OCO2 N#Cc1cc(Cl)ccc1OC(c1ccc(-n2cncn2)c(F)c1)=O c1(C(N(CCCNC(CCc2scc(C)n2)=O)C)=O)cc(C)nc(C)n1 N1(C(C2(CNC(C(CSC)O)=O)CCC2)=O)CCCC(C(N)=O)C1 C1(C(N(CCCNC(c2nc(=O)n(C)[nH]2)=O)C(C)C)=O)CN2CCN1C(C)C2 c1(C(=O)NCCCN(C(C2(CC=C)CC2)=O)CC)cccc(C2CC2)c1F CC1=C(C(=O)N2CC3(CC3C(=O)NCc3ccc(F)nc3F)C2)CCO1 CCCCCC(CCCCC)CC(=O)NCC1CCN1C(c1coc(N(C)C)n1)=O N1(C(c2n(C)ncc2)=O)CCC(C)(CCC(=O)NC2(C)CC2)C1 C(C(CNC(=O)C(F)(F)C1(O)CCC1)C(F)(F)F)NC(C1CCCCS1)=O CCCC(C#N)C(=O)N1CCC(NC(C2CC3(CCO2)CC3)=O)CC1C N1(C(C=CSC)=O)CCC2CN(C(=O)Cc3ncoc3C)CC2C1 N1(C(C2(CC#C)CC2)=O)CC(C(N2CCCC2C(C)C)=O)C(C)(C)C1 N1(C(C(C)C2=CCCC2)=O)CCC2(CC1)CCN(C(=O)COC1CCCCC1)C2 c1(CN(C(C)C)C(=O)NC(C)C(C)C)cc(I)ccc1F N1(C(C(C)C2CCC2)=O)Cc2[nH]nc(C(=O)NCC(C)(C)OCCO)c2C1 c1(C(=O)NCC(C)CNC(=O)C=CCl)cccc(-c2ccn(C)c2)c1 C12(C(=O)NC(C(=O)OCC)(C)C)CC(CO)(CN1C(C1CCC1C)=O)C2 C(=O)(C1CCC2(CN(C(=O)NC(c3cc(Cl)ccc3F)C3CC3)C2)OC1)OC c1(C(=O)NCC(N(C)C(c2nccn2C)=O)C2CC2)cc(=N)[nH]cc1Br N1(Cc2c(C)occ2)CCCOC(CNC(c2cnccc2C(F)(F)F)=O)C1 n1(C(c2ccncc2)C)nc(-c2ccco2)nc1-c1cc(-c2ccco2)on1 C(=O)(CC1=CCN(C(=O)C(C)NC=O)CC1)N(C)Cc1onc(CC)n1 N1(C(c2[nH]cc(C#N)c2)=O)CC2CCCCC2(NC(=O)C=CC2CCCO2)C1 c1(C(N(C2CCC(NC(=O)C(C)(F)F)CC2)C)=O)cnn2c1OCC2 C1(NC(c2c(OC)ccs2)=O)CC2CC1CN2C(c1cnc(C)cc1C)=O Cc1ccc(C(C)C(=O)NC(C)(C)CN(C(=O)C(C)(C)N(C)C)C)s1 CC(N=c1[nH]c(=NCC2(C)CC2(Cl)Cl)[nH]c2c1COC2)c1cccc(O)n1 c1(ONC(=O)NCC2SCC(C(C)(C)C)C2)cnc2ccccc2c1 c1(SC)nnc(N2CCCC2c2cnco2)n1CC1CC(F)(F)C1 C1(CC(=O)N(CCC)CCC)CCCN1C(=O)CC(C)c1ccccc1 C1(C(=O)NCC2(O)CC(NC(C3(C(N)=O)CCC3)=O)C2)CCCCC1O C(C1CCCN1C(=O)CC(O)CN(C)C)=CC(=O)NC(c1cc[nH]n1)C n1(CC#C)c(C)cc(C(=O)NCCCCNC(c2ccc(Cl)cc2CC)=O)c1C N1(C(c2cc(OC)c(Cl)cc2)=O)CC2CCN(C(C3CCS3(=O)=O)=O)CC2C1 Cc1noc(C)c1C(C)CC(=O)NCCC(C)(C)NC(=O)CC(C)C1CCCC1 N1(C(c2c(C(C)C)noc2)=O)CC(C(=O)N2CCCO2)CCC1(C)C C1(NC(Cc2ccc(CC)cc2)=O)CC(O)CN(C(c2cnc(O)o2)=O)C1 C1(CC)CN(C(=O)Cc2ccc(Br)s2)CCN1C(C1CCC1CF)=O Fc1cccc(Cl)c1CNc1cncc(N2CCOCC2)n1.C12CC1N2 C1(CNC(CCc2cc(C)[nH]n2)=O)CCCC(NC(c2c[nH]cc2C(C)C)=O)C1 N1(C(C2CCN(C)C2)=O)CC2(CCCC2)C1C(N1CCC(C)(F)C1)=O C1(CC(=O)NC2(CCCNC(c3n(CC)nnc3)=O)CC2)CCCCC1C N1(CC=C)C(=S)NC(c2cccc(OC)c2C)C(C(=O)OC)=C1CCl C12(NC(C3CCCC3)=O)CCCC1N(C(C1C(c3ccccc3)C1(F)F)=O)CC2 c1(C(=O)NCC(N2C(c3c(C)c(Br)ccc3)CCC2)=O)n[nH]c2c1CC(C)(C)C2 c1(CNCC2OCCN(C(C(C=C)(C)C)=O)C2)ccc(OC)c(F)c1F C1(N(C(CCCCSC)=O)C)CC2CCC(C1)N2C(c1cnn2ccsc12)=O N1(C(C(CC)(C)C(F)(F)F)=O)CCC2(CC1)OCCC2NC(c1cnco1)=O c1(CNC(=O)C(F)(F)Sc2ccc(-c3ccccn3)o2)ccc([N+](=O)[O-])c(O)c1 N1(C(C2ON=C(C)C2)=O)CCN(C(c2cc3c(s2)CCCC3)=O)C2COCC12 c1(CCC)cc(N2CCCC2CNC(=O)CC2OCCC2C)nc(Cl)n1 C1(NC(C(CCC)NC(C)=O)=O)C2CCC1CN(Cc1cc(C)ccc1Br)C2 C1(C(=O)NC2CC2NC(C2CC2F)=O)CCC(CSc2ccccc2)CC1 N1(C(CSCC=C)=O)CCCC1(C)CCC(N1CC(C)(C(C)OC)C1)=O c1(C(N(CC(C)NC(C(CC(C)C)C)=O)C)=O)cc2ccccc2cc1F c1(C(C(=O)NC(C#C)CC)NC(c2cnco2)c2nn[nH]n2)cccnc1 C1(C(C)NC(c2cnn(C(C)(C)C)c2)=O)CCN(C(C2CCS2(=O)=O)=O)CC1 c1(NC(C2(C)N(C(c3cccc(N(C)C)c3)=O)CCC2)=O)cc(F)c(O)c(F)c1 C1(NCc2ccc(-c3c(OC)ncnc3OC)s2)CCc2ncccc2C1 n1(CC(=O)N(CC(CN(C(C2CCC(C)O2)=O)C)O)C)ccc(=O)n(C)c1=O c1(-c2cn(C(C(=O)NCCCCC)C)nn2)ccc2c(c1)NC(=O)C2 C1(C(N(CC#CC)C)=O)CN(C(=O)CCc2nccn2C)CC1C c1(C(C)C)ccc(C(=O)NCC2CC(F)CN2C(=O)CN2CCCCC2)nc1 c1(C(=O)NC2CCC(NC(C3C=CCCC3)=O)C2)ccn2ncc(Br)c2c1 c1(NCC(C(c2ccc(C)cc2)=O)N)cc2nc(C)cc(C(F)(F)Cl)n2n1 c1(OC)ccc(-c2nc(NC(c3cc(O)nc(Cl)c3)=O)cs2)c(Cl)c1 C1(C(=O)OC)CCN(CC(=O)N(C)Cc2cc(C)n(C)n2)C(c2cnn(C)c2)C1 C1(C)(C(N2CC(NC(CCCCC)=O)C(C)(C)C2)=O)CCCCC1(F)F C1(CC#S(=O)CCCc2ccccc2)CC2(CCNCC2)C1 c1(OC)cc(F)c(F)cc1C(=O)N(C1CC(CF)C1)C(=O)CC1(OC)CCCC1 C1(NC(=O)NC(c2nc(C(C)(C)C)cs2)C)CCCCCCC1C(F)F C1(NC(CC(C)=CC)=O)(CO)CCN(C(c2ccc(O)cc2OC)=O)CC1 c1(CC)cc(C(N2CCC(C(=O)Nc3cc(C(F)F)ccc3F)C2)=O)cc(C)n1 c1(NC(C(C(C)C)C)CNC(C2(C)CCCCC2)=O)c(C#N)cccc1[N+](=O)[O-] C1(COCC(N2CC(CNC(=O)CC3CCOCC3)C2)=O)C2CCC3C(C2)CC13 N1(C(C2(C#N)CC=CC2)=O)CC2CCOC2(CNC(C2CCC2)=O)C1 C1(CNC(C(F)=CC)=O)(NC(=O)COC(C)(C)CC)CCCCCC1 c1(CNCc2ccc(-c3cnc(=N)[nH]c3)cn2)c[nH]c2cccnc12 C(=O)(CC(C)C(=O)c1ccccc1)N(c1ccccc1C)CC c1(C(N2CC(NC(CC3CC(=C)C3)=O)C(SC)C2)=O)ccc(=O)n(C2CC2)c1 CC1CCN(C(N)=O)CC1CC(=O)NCC1CC(NC(=O)COCC2CCCO2)C1 c1(CCC)nc(C)c(-c2nc(CCc3ccncc3)nn2-c2cccc(Cl)c2)s1 C(CC(C(C)(C)C)NC(C1COCC1C(N)=O)=O)N(C(C(COCC)(C)C)=O)C C(=O)(C(CCN(C)C)N(C)C)N(CC(=O)NCc1n(CC)cnn1)C Cc1ccc(F)c(C(=O)N(C)CC2CCCC2NC(C2(CF)CCOCC2)=O)n1 C=CC1(CC(=O)NC2CSCC2C)CN(C(=O)CCC2CCCC2)C1 c1(C(=O)NC2CC(NC(c3ccc(CC)s3)=O)C2)ccccc1C(C)O C1(CNC(c2coc(C(F)F)c2)=O)CC(O)CN1C(C1CCCC1C(F)F)=O Cc1noc(C2CC2)c1C(N1CC(NC(c2cnn(C3CCC3)c2)=O)C(C)C1)=O C1(NC(c2c(CC)n(C)cc2)=O)COC2C(NC(=O)CC3CCCOC3)COC12 Cc1nn(C)c(C)c1CCC(=O)NC(C)(CNC(C1CCCC(F)C1)=O)C1CC1 C1(CCNC(c2cncnc2)=O)CN(C(=O)Cc2cccc(O)c2)CCS1(=O)=O C1(CC(=O)NCC(CC)N(C(=O)CNC(N)=O)C)CCCCN1C c1(OC)cc(CN2CCC(C(C)NC(c3ccc(O)nc3)=O)CC2)ccn1 Cc1nc(N2CCN(C)C(CNC(=O)CC3CCCC4(CC4)C3)C2)cc(O)n1 c1(CNc2cc(OCC(C)C)ncc2)cc(Cl)cc(C#N)c1 N1(C(CC(CNC(C=C(C)C2CC2)=O)C)=O)CCn2c(C)cnc2C1 C1(NC(C(C(C)C)C2CCC2)=O)CC2CCCC(C1)N2C(C1CC(O)(C#N)C1)=O c1(C(=O)NC2CCN(C(C(CC#C)C)=O)C2)cccn(CC(F)(F)F)c1=O c1(CCCNC(c2ccc(Cl)c(Cl)c2)C(=O)OCC)nnc2n1CCCC2 c1(OC)ncc(NC(c2cnc(CNC(=O)CC3CCCC3)nc2)=O)cc1C C1(C(=O)NCC2C3CN(C(C4N(CC)CCOC4)=O)CC32)CC12CCCCC2 N1(C(C(C2CN(C(c3ccc[nH]3)=O)C2)OC)=O)CC2CCC(C1)O2 S(=O)(=O)(c1ccc(NCC2CCCCN2C(C)(C)C)cc1Cl)NC1C(C)C1 CC(C)C(C)C(=O)NCCOC1CN(C(=O)CCN2CCCS2(=O)=O)C1 C1(NC(C2C(C)CCO2)=O)CCN(C(c2ccc(C(C)(C)C)s2)=O)CCC1(F)F C1(C(C)C)(C(=O)NCC2CN(C(=O)COCc3nc[nH]n3)CCO2)CC(C)(C)C1 C(C(C(C)(C)C)NC(=O)CCC1CC1)NC(C1CC(C(F)(F)F)(OC)C1)=O CCCC(C)(C)CC(=O)NCCCOCCCNC(C1CCN(C)C1CC)=O N1(C(c2nc(CC)oc2)=O)Cc2[nH]nc(C(=O)N(C3CCSC3)CC)c2C1 N1(C(C(C)Oc2ccc(OC)cc2)=O)CCC2(CC1)CC(=O)NCC2O C(=O)(C(C(=O)N(C(C)(C(=O)Nc1cccnc1C)C1CC1)C)OC)OC C1(C(=O)NC2CCC(C)N(C(=O)Cn3nccn3)C2)CCc2ccnn2C1 C1(NC(COc2c(OC)cccc2)=O)(CO)CCN(C(c2n[nH]c(=N)[nH]2)=O)CC1 C1(c2n(CCCSCC)nnn2)(NCc2cn(CCO)nc2C)CSCCSC1 CC1CCN(C(=O)C(C)(C)F)CC1NC(c1n[nH]cc1C(F)(F)F)=O N1(C(C(C)CF)=O)CCCCC1CNC(=O)Cn1nnc(=O)[nH]1 C1(CC(=O)NC(CCNC(c2c(C(=O)OC)coc2)=O)C)C(=O)N(C)N=C1C C(C(C(C)C)C(C)C)(c1n(-c2c(CC)cccc2)nnn1)NCC1(C)CC1(C)C C1(C(=O)NC2CCC(NC(C(C)C3CC3)=O)C2)CC2(CSC2)C1 N1(C(CC(CCC)(C)C)=O)CCC2(CC1)CN(C(=O)C1=NOC(C)C1)C2 n1(CCC(=O)NCCN(C(C(CC)C)=O)CCCN(C)C)ccc(O)nc1=O N(C(=NCCCCC(F)(F)F)NCCCCc1ccc(Br)cc1)C1CC(C)SC1 C1(CC(=O)NCCCN(C)C2CC2)CCN(C(c2ncccc2F)=O)CC1 c1(C(=O)NCC(C2CCC2)NC(C2C(=C)C2)=O)c[nH]cc1-c1csc(C)n1 CC1CC(C(N2CCCC(CC3CC3)C2)=O)CN(C(C2(Cl)CC2)=O)C1 c1(C(=O)NC2CC(C)(NC(C=C3CCC(C)C3)=O)C2)c(C(F)(F)F)ncn1O C1(CC)CN(C(C2CC(O)C2)=O)CC1C(=O)Nc1ccc(F)cc1 C(CN=C(NCC(C1CC1)OC)NC(c1cccs1)C)c1onc(CC)n1 C1(C(=O)NCC2CCN(C(Cn3ncc(C#N)c3)=O)C2)C(F)(F)C12CCC2 Cn1cnc2c1CCCC2C(=O)NCC(CO)NC(=O)C(C)(C)c1ccnn1C C(F)(c1ccccc1)=CC(=O)NCC(CCOC)NC(=O)C(c1nc(C)cs1)C c1(C(NNC(=O)NCc2scc(SC)c2)=O)ccc([N+](=O)[O-])c(C)c1 c1(NCc2c(NC(=O)CCC(C)N(C)C)ccc(C)c2)[nH]cnc2nc(Br)cc1-2 C(C(C)C(F)C(=O)N1CCCC1COC)NC(CC=C=C)=O c1(CN(C2CC(N)C2)C(c2ncc(OC)cn2)=O)cc2ccncc2[nH]1 c1(C(N2CCCC(Nc3nccc(C(=O)OC)n3)C2)=O)ccc2n[nH]cc2c1 c1(N2CCC(NC(C(CC)n3cncn3)=O)C2)ncc2ccsc2n1 Cc1cc(C(=O)NC2CC2c2ccn(-c3ccccc3)n2)nc(C)c1 N1(S(C)(=O)=O)CCCC(CC(=O)NCC(C2CC2)NC(=O)Cc2ccon2)C1 C1(CNc2nc(SC)c(F)cn2)CCC2(CCN(C(=O)C(F)(F)F)CC2)O1 C1(C#N)(C(N2CC=CC(C(N3CC(N(C)CC)C3)=O)C2)=O)CCCCC1 C1(CCCNC(CCC=CC)=O)CCN(C(c2sccc2COC)=O)CC1 CCC(C)(C(=O)OC)NC(C1CC=CCN1C(=O)CC1C(C)(C)C1(C)C)=O C(=O)(C(=O)NCCN1CCCC1)NCCN(C)C CC1CCC(=CC(=O)NCC2CCN2C(C2(C(F)(F)F)CC=CCO2)=O)CC1 N1(CC(C)C)CCC(C(N2CCN(C(C3COC(C)C3)=O)CC2)=O)CC1 N1(C(C(C)OCC2CCCCO2)=O)CCC(F)C(NC(c2c(Cl)nsc2Cl)=O)C1 C1(CNc2ncnc(=N)[nH]2)CS(=O)(=O)CC1NC(=O)CCOC1CCCCC1 Cc1[nH]c(C(=O)NC(c2ccccc2)C#N)c(C)c1C(N1CC2CC1CN2C)=O O(NC(=O)C(C)NC(c1ccc(NC)cc1)=O)CC(=C)Cl C1(CC)CN(C(=O)CN(C(=O)CCc2nncs2)C2CCC2)CCN1C C1(NC(C(CCC)C)=O)CC2(CCN(C(c3ccc4c(n3)NCC4)=O)C2)C1 C1(Cn2cc(CN(C)CC)nn2)CCCCN1C(=O)Cc1cn(CC(=O)O)nn1 c1(C(N2CC(O)(CNC(CCCC=C)=O)C2)=O)cc(F)cc(C)c1N c1(C(=O)NC2(C)CN(C(C(CC)O)=O)C2)ccc(C(=O)OC)n1C N1(C(C(c2ccc(OC)cc2)CC)=O)CC2OCCN(C(c3ccoc3)=O)C2C1 c1(NCC2OCC(COC)C2)cc(=O)n(C)cn1 C12(CNC(c3ccc(OC)s3)=O)CC1CN(C(C1CCS1(=O)=O)=O)C2 c1(C(=O)NC2C(CC(=O)N(CCC(F)(F)F)C)C(O)C2)cn(C)ccc1=O C(=O)(C#CC(C)(C)CNC(=O)C(C=C)OC)N1C(CC=C)CCCC1 C1(NC(C2(CC)CNC(=O)C2)=O)CCCCCC1NC(=O)Cc1cc(OC)no1 C=CCC(CC(=O)NC(CCO)C(C)(C)C)NC(=O)C(C)(C)C=C C1(C(N2CCC(C(C)(C)C(=O)NC3CC3c3cncs3)C2)=O)CC(N=[N+]=[N-])C1 Cc1cc(N)ccc1C(=O)NC1CC2(C1)CC(NC(=O)C(C)c1cccs1)C2 c1(C(=O)OC)cc2c(nc1NC1CCCN(C(=O)C(C)CC3CC3)CC1)CCC2 Cn1nc(C(=O)NC2(CNC(=O)CC3CC(=O)C3)CC2)c2c1CCSC2 N1(C(C(C2CCCC2)C)=O)CC2CCOC2(CNC(c2ccn(C(F)F)n2)=O)C1 n1(CCC)cc(C(=O)NCCCNC(=O)C(O)C(C)c2ccccc2F)c(C)n1 c1(CC)oc(C(=O)NC(C)(CNC(=O)Cc2ccc(Br)cc2)CC)cc1C CN1CCN(C(C2COCCN2CC(F)F)=O)C(CNC(C2CC3(CC3)C2)=O)C1 CC1CCc2nc(C(N3CCC(C(=O)O)(CO)CC3)=O)cn2C1 N1(C(C2CN(C(CC#N)=O)C2)=O)CCCCC1CO C1(C(N2CCCC(CCCC)C2)=O)C2CC3C(C2NC(C2(Cl)CC2)=O)C13 C1(C(N2CCC(CN(C(=O)CN3C(=O)CCC3=O)C)C2)=O)CC(C2CCC2)C1 CCCC(CNC(=O)CCCCNC(C)=O)C(=O)N(C)CC1(O)CCCCC1 N1(C(C)=O)CC2CC2(C(=O)NC(C)CN(C(=O)CCc2nc(O)n[nH]2)C)C1 N1(C(C(=O)NCCCSC)C2CC2C)CCCC(C)(C)C1 C12CCCCN1C2=O.C12(NC(=O)NCC)CCC(C1)OC2 C12CCCCCN1C2=O.C12(C(N(C3CCOCC3)C)=O)CCCC1C2Br C(C)(C)(CCC(=O)NCCCCO)NC(C=CC(CC)C)=O C1(CNC(c2c(C)nc(O)[nH]2)=O)C(C2CC2)CCN1C(=O)CCC1(C)CC1 C(=O)(CCC(C)(C)C#N)N1C(CCNC(C(C(C)C)CN(C)C)=O)CCC1 C1(C(=O)NC(c2cn(C)nc2)CO)C=CCN(C(c2cnnn2C)=O)C1 N1(c2nccc(NC(CCn3ncc(C)c3)=O)c2)CC(C)OC(C)C1 C1(NC(C(Cc2ccco2)NC(=O)CCc2cccs2)=O)C2CCCC1COC2 C1(NC(C2CCOC2)=O)CCCCC12CCN(C(c1n[nH]cc1Cl)=O)CC2 C(=O)(C1CCCc2cc(O)ccc21)N1CC(N(C(c2c(COC)cco2)=O)C)C1 c1(NC(C2(Cc3ccccc3)CCNC2)=O)cncc(OC)n1 c1(SCC(=O)N(CC(C)NC(=O)Cc2cscc2Br)C)ccccc1 CCCC(C(=O)NC1CCN(C(c2cncnc2C(C)C)=O)C1)NC(N)=O Cn1c(C(N2CC3CCCC3(NC(C3CCC(O)CC3)=O)C2)=O)cc2sccc12 C(=O)(C1=CCC2CCC1N2C(c1ccc(C)s1)=O)NC(CC)C(C)(C)C c1(C(N2CCC(OC)(CNC(=O)CSCC(C)C)CC2)=O)ccc(C)c(C)c1O N=c1[nH]nc(C(=O)NCc2ccoc2C(F)(F)F)s1 C1(CNC(C(CCSC)OC)=O)CN(C(=O)Cc2cc(C)ccc2F)CC1(C)C c1(C(=O)NCCN(C(CC=C=C)=O)CC(C)O)cc(F)cc2c1NCCC2 c1(C(=O)N)nccc(OC)c1N.c1(COC)cn(C2COC2)nn1.C12CC1C(=O)NC2 C(C(C)C)(C(O)C(=O)NC(C(=O)NC(CC1CCCC1)CO)C1CCC1)OC N1(C(C(CCCC)F)=O)CCC(C=C)(C(=O)NC(C2CCOC2)CC)CC1 c1(OC)cc(CCNC(=O)CCCC(=O)N(C)C)cc(OC)c1OC(F)F CC(CS(C)(=O)=O)C(=O)N=c1cc(C2CCOCC2)[nH][nH]1 C1(C)(C(=O)NC(C2CCN(C(c3cn(CC)nn3)=O)C2)C)CCCN(C)C1 c1(C(N(CCN(C(=O)CC2CC2C)C(C)C)C)=O)c(C(F)F)cccc1F N1(C(c2c(OC)cc(F)cc2)=O)CCCC(C2(NC(=O)C(C)=CC(C)(C)C)CC2)C1 CC(C)C(C(=O)NCC12CCC(CC1)N2C(c1ncccc1N)=O)C(C)C C=C=CCCC(=O)NCCn1ccc(C(=O)NCC(C)(O)CSC)c1 N1(C(c2cc(CC)n(C)n2)=O)CC(C(=O)NC2CCN(CC)CC2C)CC(C)C1 c1(C(N(CCNC(C2CC(=C)C2)=O)CC)=O)c(Br)ccc(OC)c1C C(=O)(CCCCCCCC1CC1)NC1CCN(C(c2cnc(C)s2)=O)C1C1CC1 N1(C(Cn2c(C)ccn2)=O)CC2CCC(C1)N2C(C1CC(F)C1)=O CC1CC(C(=O)NCCCCCNC(c2cc3n(n2)CCCC3)=O)CC(C)(C)C1 C(=O)(C(C)(C(F)F)c1ccccc1)NC1C(C)CN(C(=O)Cc2cccnc2)C1 C1(C)(NC(c2ccnc(C)n2)=O)CCCN(C(c2ccc(C)c(F)n2)=O)C1 Cc1ccc2nc(C(=O)NC(C3CCCCN3C(=O)CC(F)F)C)ccc2c1 C(=O)(C1(C)CCn2ccnc21)N1CC2(C(NC(Cc3c(C)nccc3)=O)CC2)C1 C1(C(=O)OC)CN(C(=O)NC2CCCC3(CCOC3)O2)CC12CCCCC2 N1(C(CCCC#CC)=O)CC2CCC(NC(=O)Cn3ncc(O)nc3=O)CC2C1 c1(C(=O)NC2CCC(F)(F)C2)c(F)ccc2ccoc12 C(=O)(C(CC(C)C)C(N)=O)NC1CCC(CC(=O)N(CCOC)CC2CC2)CC1 C1(CNC(c2ccnnc2O)=O)CC2(CCN(C(C3(F)C4CCCC34)=O)CC2)C1 CC(CC(C)(C)C)C(F)C(=O)NCC=CCNC(c1ccnc2[nH]ncc12)=O C1(C(=O)NCC2(C)CCN(C(c3cnc(C)s3)=O)C2)C2Cc3ccccc3C12 C(N=c1[nH]c(N2CCc3[nH]nc(O)c3C2)nc2ccsc12)c1c(O)nccc1 C1(C(C)(C)C)CN(N2CC3(CC(C)CC3)C2)CCO1 c1(OCC(C)C)cccc(-c2ncsc2C(=O)NCCc2ccncc2Br)c1 c1(OC(C)C(=O)N(C2C3CN(C(c4n[nH]c(=N)s4)=O)CC23)C)ccc(F)cc1 C(=O)(CC(CC)C(C)C)N1C(C(N(CC(=O)OC)C)=O)C2CCC1C2 N1(C(c2n[nH]cc2F)=O)CCCc2ccccc2CC1 C1(C(=O)N(C(C(=O)N(CCNC(=O)NCC)C2CC2)C)C)CC(F)CN1C.CSC c1(OC)ccc(CN2CCC(C(N3CCOCC3)=O)C2)c(Cl)n1 Cc1nc2cccc(C(=O)NC(C)CC(C)Nc3ncc4c(n3)CCCC4)c2[nH]1 c1(OC)cccc(SCC(=O)NC2CCC(NC(C3(C)CC3F)=O)CC2)c1 C1(CNC(C2CC(OC)CC2C(F)F)=O)COC2(CCC(C)CC2)O1 C=CC(C)C(C)C(=O)N(CCC)CCNC(c1cc(Cl)ccc1C)=O c1(CC(=O)NC2CN(C(CSCCOC)=O)CC2CO)c[nH]c2ccc(Cl)cc12 c1(C(N(C(C)C)CCN(C)C(c2cccnn2)=O)=O)cc(Br)cnc1O C1(CC)CC(O)CCN1C(C1CCN(C(c2c[nH]cc2C2CC2)=O)C1)=O C(=O)(CC(F)(F)C(F)F)NCC1OCCN(C(Cn2c(C)csc2=O)=O)C1 CN1CCC(C(N2CC(C(N3CCCOC(CCO)C3)=O)C(C)(C)C2)=O)CC1=O O=C1CCC(C(N2CCC(C(=O)Nc3ccc[n+]([O-])c3)CC2)=O)CN1 c1(CCC)cc(NC(C)(CC(C)CC)c2nnnn2C2CC2)cc(C)c1 S(=O)(=O)(c1cnn(C(C)C)c1)N1CCCC(CC(C)C)C1 N1(C(c2ncn(CC)n2)=O)C2CCC1CC(N(C(=O)CC1COC3CC1C3)C)C2 c1(OC)ccc(CN2CCN(C(=O)OC)C(C)C2=O)cc1Br Cc1cccc(C)c1CNC(=O)CC1CC(NC(C2CCC(=O)NC2)=O)C1 C12(C(=O)NCCC(CC)C)CCC(CN(C(=O)C=Cc3cnn(C)c3)C1)C2 c1(C(N2CCCC(C(=O)NC3N(C)C(=O)NC3)CC2)=O)cc2ccsc2n1C C(N=c1[nH]c(=NCCOc2ccc(Cl)cc2)[nH]c2c1COC2)c1c(C)cn(C)n1 N(C1CCC(C)(C)c2cc(Br)ccc21)C(=O)NC1Cc2c(C)[nH]nc2CC1 CC(C)CC(C(=O)NC(c1ccco1)CO)ONC(C12CCCN(CC1)C2)=O C12(C(=O)NCC3(O)CC3)C3CC1C1C(C(N4CCCC(C=C)C4)=O)C3C21 C1(CN(C(CC)C(=O)OC)C(=O)CNC(=O)CN(C)C)CCCCC1F Cc1nc(NCc2ncc(CO)o2)cc(N(CCC(F)(F)F)C)n1 c1(SCC(N2CCC(N(C(c3ncoc3CC3CC3)=O)CC)C2)=O)cccc(F)c1 N1(CC(=O)NC(C)CN(C(=O)C(c2cnccn2)C)C)CCC(=O)NC1=O C1(c2cn(CCN(C(=O)CC(O)c3cnc(Cl)s3)CC)nn2)CCCCCC1 N1(C(C2(F)C(C)C2)=O)CC2OCCN(C(=O)C(F)F)C2C1 Cc1cc(C)c(C(=O)NC2CCN(C(c3ncoc3C)=O)CC2C)c(C)n1 C1(CC=C)(NC(=O)C(CC)OCC)CCCN(C(=O)CC(Cl)Cl)C1 N1(C(C2CN(C(C(CC=C)OC)=O)CC(C)O2)=O)C(CO)CCC12CCC2 C(CNC(c1c(C)oc(C)c1C)=O)(C(C)C(C)C)NC(CC(=O)NCC)=O Cc1c[nH]c(C(N2CCCC(N(C(=O)CSCc3ccccn3)C)C2)=O)cc1=O NS(=O)(=O)c1csc(C(=O)NCC2CN(c3ncncc3Cl)C2)c1 c1(C(=O)NC(C)C(C)NC(c2cccs2)=O)sc2sccc2c1Cl C(C(C(=O)NCC(O)C(F)F)n1cc(Cn2cccn2)nn1)OCC C1(CNC(C(C(C)C)SCC)=O)CCN(C(c2sncc2C)=O)C1(C)C c1(N(C)C)cc(C(=O)NC2CCOCC2NC(C23CCCC2C3)=O)ccn1 c1(CCCC)cc(C(=O)NCc2ccccc2O)c(C)o1 c1(C(=O)NCC(C)(O)CNC(C2CC(F)C2)=O)cc(C#N)cs1 c1(OCC)cc(C(N2CCC(N(C(=O)C(C)C(C)C)CCO)CC2)=O)oc(=O)c1 N1(C(C=CC=CCCCCC)=O)CC2CCC(C(=O)OCC(CC)OC)C2C1 c1(CNC(C(C(C)NC(C(c2ccn(C)c2)C)=O)C)=O)cc(C#N)n(C)n1 C1(c2cc(C)[nH]n2)CCCCN1C(=O)C(N1CCCC(C)C1)=O.CCC=O c1(NC(C2(C)N(C(C(C)OC3(C)CC4CC4C3)=O)CCC2)=O)cc(N)cc(F)c1 c1(CC)noc(CCCC(=O)NCC2CCN(C(=O)CCCC3CC3)C2)n1 N1(c2sccc2)CC(NC(=NCC2CC3CCC2O3)NCC2CC2)CC1=O C1(NC(=NN(CC=C)C(C)C)NC2CCCC2)CCCC2(CCC(F)(F)CC2)O1 CC1CN(C(c2ncoc2-c2ccon2)=O)CCC1N(C(=O)CCC(N)=O)C C1(C(=O)NC2C(NC(C3(C)CCN(C)C3)=O)C2)CC2(CCCCC2)C1 c1(C(CC(=O)NCC(O)CF)C)c(F)cccc1Br N1(C(Cc2cnc(C)s2)=O)CCC(CNC(C2CCCC(=O)N2)=O)C(F)(F)CC1 c1(C(N2CCCC(NC(C3CC4CCC3C4)=O)C2)=O)cc(F)ccc1F C1(CNC(C(c2c(C)nccc2)C)=O)CC2CCC1N2C(=O)C(F)=CCCF C=CCC(CNC(C1C=CCN1C(c1cnn2c1OCC2)=O)=O)CC(C)C c1(C(C)(C)C)cccc(SCC(N2CC(CO)(NC(C3(C4CC4)CC3)=O)C2)=O)c1 C(C(C(=O)NCCC(C)(C)N(C)C)C(C)C)NC(C(C)=CC1CC1)=O N1(C(CN(C2CCS(=O)(=O)C2)C)=O)CC2CCC1C(C(=O)N(C)C1CC1)C2 CCC(F)(F)C(C)(C)C(=O)N1CCCC2CN(c3cccc(F)c3C#N)CC12 C1(C)(NC(c2c(OC)nc(C)cc2)=O)CCOC12CC2(F)F c1(C(=O)NCC2CN(C(C3CC3F)=O)CC23CCC3)cccc2cc(F)ccc12 C1(NC(C(CC)(CC)CC)=O)CCC2CN(c3ncc(O)cn3)CCC2C1 N1(C(C(C)C(C)(F)F)=O)CCC2(C1)CN(C(c1cc[nH]c3nccc1-3)=O)CCO2 CC(C)CC(C)CC(C)C(=O)N1CCCC1C(C)(C)NC(C1CC12CCC2)=O c1(C(=O)NC2CCC(NC(Cc3nc(=N)[nH][nH]3)=O)CC2)ccc(C2CC2)c(F)c1 C1(CNC(c2cc(C)oc2C)=O)CN(C(=O)C#CC(=O)N(C)C)CCCO1 O=C(C#CCNC(C1C2CCC(C2)C1CO)=O)NOCCCC1CC1 C1(C(=O)NCC2C(C(=O)NCc3[nH]nc(CC)n3)OCC2)CCCN(C)C1 C1(NC(C2CCC(CCC(=O)OC)O2)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC1 C1(NC(c2cn(CCC)nc2)=O)CCN(C(=O)CCc2cnn(C)c2C)CC1C c1(C(N2CC3(CC(NC(C4CCC(OC)C4)=O)C3)C2)=O)cc2c(Cl)cncc2s1 C1(NC(CC(C)C)=O)CCC(C)N(CC(C)C(F)(F)F)C1 C1(NC(CCC(=O)NC(C)C)=O)CCN(C(=O)CC2COCC(C)(C)O2)C1(C)C c1(OC)cccc(NC(=O)C(=O)OC)c1.c1(CC(C)O)noc(SC)n1 N1(C(C(C)OCCC#C)=O)CC2(C1)CN(C(=O)C=Cc1c(C)noc1C)CCO2 C=CCC(C)(CC)C(=O)N1CCC(C)(CNC(=O)CC2(C#N)CCOCC2)CC1 CC(C)CCCOCC(N1CCCC1C(C)NC(=O)C(N1CCCC1)C1CC1)=O C1(C(N2CC(C(C)NC(=O)C3=CCC3)C2)=O)CCc2cc(Br)ccc2O1 c1(C(=O)NC2CC(NC(=O)CN3CCC(CO)CC3)C2)ccc2nccnc2c1 C(=O)(C(C(C)(C)C)NC(=O)COC)NCC(CC=C)(C)C CC12CC(C(N3CCCC(NC(C4CCCC(F)C4)=O)C3)=O)(C1)C1(CCC1)O2 n1(CC(=O)N(C2CN(C(=O)CCC(=O)N(C)C)C2)CC)ncn(C)c1=O c1(CC(=O)NC2CCN(C(CC3N(C)CCC3)=O)C2)cc(F)cc2c1OCOC2 C1(C(=O)NCC(CNC(=O)Cc2c[nH]nc2O)O)CCc2n[nH]cc2C1 N1(C(Cc2cnc(C)o2)=O)CC(NC(=O)CCNC(c2ccncc2)=O)C(C)C1 C1(CNC(=O)CC2CNC(=O)C2)C(O)C(O)CN1C(=O)C=C1CCCCC1 c1(C(C)OC2CCCCC2)nc(-c2cccnc2)nn1Cc1cccs1 C(CCCCCCO)NC(C1C(O)CCN1C(c1cc(I)ncn1)=O)=O Cn1[nH]c(=NC(=O)CSc2nc(-c3ccc(Cl)cc3)no2)cc1C1CCCC1 C1(NC(C2(CCOC)CC2)=O)CN(C(C23COC(CCO2)C3)=O)CCC1C C1(NC(c2c(CC)onc2)=O)CC(F)CN(C(c2cccc(O)c2F)=O)C1 C(CC(CC)C(=O)NCC(O)CNC(c1ccnc(OCCO)c1)=O)=CC c1(C(N(C2CCCN(C(C3(C)CCSCC3)=O)CC2)CC)=O)cc(Cl)ccc1F N1(C(CCOC)=O)CCC2(CCCN(C(c3ccc4c(c3)OCCN4C)=O)C2)C1 CCCCCCCCCC(C)CC(=O)N1CC2(CCN(C(=O)CCS(C)=O)C2)C1 n1(CC(=O)NC2C(CNC(C(c3[nH]c(=N)sc3)=O)=O)CC2)cnc([N+](=O)[O-])n1 C1(NC(C(CC)SC)=O)CC2CC(C1)N(C(c1cc(C3CC3)ncn1)=O)C2 c1(C(N(C)CC2CC(F)CN2C(=O)Cc2cn(C)nn2)=O)nccc2[nH]ccc12 c1(NC(=O)NC)cccc(C(=O)NC2C(C(=O)O)CC2)c1.C(=O)(C(O)CC)NCCO O=C(C1=CS(=O)CCC1)NC1(CNC(c2cc(C3CC3)ccc2F)=O)CCOC1 Cc1nc2cc(C(=O)NC3CC(C)(NC(C4CC4C)=O)C3)[nH]c2s1 C1(C)(C(=O)NC(C(C)C)C2(c3cccnc3)CCC2)CCC(=O)N(C)C1 C1(C(=O)N(C2CCCC2)CCCNC(=O)CCCC2(C)N=N2)(OCC)CCOC1 N1(C(CNC(N)=O)=O)CCC(O)C1C(N1CCC=C(Cl)C1)=O c1(C(N(C)CC2(CN)CCC2)=O)ccccc1CO c1(C(N2C(CNC(c3cc(CO)ccc3Cl)=O)C=CC2)=O)cc2ccccc2s1 c1(C(N(CCN(C(C)C)C(c2ccc(CCCCCO)o2)=O)C)C)ccccc1Cl C1(NC(c2c(C)scc2)=O)C2CC(CN(C(c3cc(Cl)no3)=O)C2)C1CO C1(NC(C2(C=C)CCC2)=O)CC2CCC1(CNC(=O)C(C)(C)C1CCCC1)C2 C1(C(=O)NC(CC)C(C)CN(C)C)CC2CC1CN(C(c1n[nH]c(C)c1O)=O)C2 C(=O)(CCN=C(NCC(C)(C)c1ccsc1)NC1CCN(CC2CC2)C1)NC C1(NC(c2nccc(CC)c2)=O)CC(O)CN(C(c2c(C)cncc2C)=O)C1 C12(C(N3CCC(CNC(c4c(N)c(Cl)ccc4)=O)C3)=O)CC1Cc1c[nH]nc12 c1(OCC(C(=O)NC2CCN(c3ncc(C)cn3)CC2F)OC)ccc(F)cc1F N1(C(c2cc(SC)oc2)=O)CCC(F)(CNC(C2CC23CCOCC3)=O)CC1 N1(C(C(C)Oc2ccc(F)cc2F)=O)CC2CN(C(=O)C3=CCCCC3)CC2C1 c1(C(=O)NCC2CN(C(c3ccn(C)c3)=O)C3C2C3)cc2sc(Cl)cc2s1 C1(C(N2CC(C)(NC(c3ccc4cncn4c3)=O)C2)=O)CC2CC1C1C2C1(F)F CCC(C)CCC(=O)N1CC2(CC(NC(c3ccccc3CC#N)=O)C2)C1 C(C)(C)(C(c1nnnn1C(C)C(=O)OC)NCc1noc(C)n1)OC N1(C(c2ncn(C(C)C)c2)=O)CCCC(F)(C(=O)NCc2ccnc(Cl)c2)C1 c1(CC)csc(S(=O)(=O)NC(C)C(C(=O)OC(C)C)OC)n1 N1(C(C(C)OCC(C)C)=O)CCC(C)(CCNC(C2CCNC2=O)=O)C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CCC(NC(c3ccsc3)=O)(C2)C1 c1(C(=O)NCCC2(C)CCN(C(C(C)OCC=C)=O)CC2)ccc(S(N)(=O)=O)s1 C1(C(C)NC(=O)C(c2cncn2C)C)CCCN(C(c2cn[nH]c2)=O)C1 N1(C(C2CC(C)S(=O)(=O)CC2)=O)CCN(C(=O)C2=CS(=O)CCC2)C2(CCC2)C1 C1(CCOC)(NC(C2CC=CCO2)=O)CCN(C(=O)COc2cccc(Cl)c2)C1 C12(C(=O)NCCCCCNC(=O)CC3CC3C(F)(F)F)CC=CC(C1)OC2 CC1CCN(C(=O)CCc2cccn2C)CC1CC(=O)NCCC1CCOCC1 N1(c2nccc(NC=O)c2)CC2C3CCC(CC3)C2C1.CC(C)C c1(C(N2CCC(C(C(C)C)NC(CCC)=O)CC2)=O)nccc2ccsc12 C1(NC(CC(CC)CN(C)C)=O)CN(C(=O)Cc2ccco2)CC2(CC2)C1 C(C(C)(COC)C(=O)NCCCCCC(=O)NC1(C)CCC(C)CC1)OC C(=O)(C(C)(C)C)NC(C)CCN(C(c1[nH]nnc1-c1ccnn1C)=O)CC c1(C(=O)NC2CCCN(C(C(C#C)(C)C)=O)CC2)[nH]nc2ncccc12 CC1=C(C(=O)NC2(C)CC(NC(=O)CCc3ccnn3C)C2)C(C)(C)CCC1 C1(C(C(C)C)NC(=O)C(n2cc(Cc3ccsc3)nn2)C)CCOCC1 C1(NC(CCCCOCCC=C)=O)CCN(C(=O)C=CCCC)CC12CCC2 CC(C)C(F)(F)CC(=O)NCC1CCCN(C(c2cnsn2)=O)CC1 C1(C(C)C)CC(C)CN(CC=O)C1.c1(Cc2nnnn2C)cnn(C)c1C Cc1ccc(C(N2CCC(Cc3cc(F)ccc3F)CC2)=O)c(O)c1 c1(C(=O)NCCCCC2(NC(=O)CC3CCC3)CC2)cscc1Cl c1(C2C(=O)N2C(C)Cn2cnnc2)cccnc1.c1(CC(=O)OC)cnsc1 N1(C(C2C(OC)CCC2)=O)C2CC1CN(C(c1ncc(F)cn1)=O)C2 C=CCC(CC)C(=O)NC(CC(=C)C)C(=O)NCc1ncccc1C N1(Cc2c(C)ccs2)CC2(CCC(CNC(c3ccc4c[nH]nc4c3)=O)O2)C1 c1(CSC(C(=O)C2(C(=O)NC(C3(C)CC3)Cl)CC2)SC)ccc(C(C)=O)cc1.OC Cc1cc(Br)nc(Cl)c1NC(C1CCCC(=O)C1)=O c1(CCNC(=O)NCCCSc2ccccc2)sc(Cl)cc1Br c1(NC(=O)NC2C(SC)CCC2)cnc(C)nc1C C1(NC(C(C2CC(NC(CNC(C3C(C)C3)=O)=O)C2)F)=O)CN2CCCC1C2 c1(CCC)ccccc1C(=O)NCC(C)NC(C1(C(F)(F)F)CC(O)C1)=O C1(c2n(CC)nnn2)(NCC2C(C)C2C)COc2ccccc2SC1 c1(C(=O)NCC=CCNC(C2CC(C)(F)C2)=O)cncc(-c2ccoc2)c1 N1(C(C2OCC(C)(C)OC2)=O)C2CCC1CN(C(=O)C1=CCCCCC1)C2 c1(C(N2C(CNC(C(C)n3cncn3)=O)C=CC2)=O)ccc(N(C)C)nn1 N1(C(c2cc(C)cc(Br)c2F)C(=O)NC)Cc2ccccc2C(CO)C1 C=C(C)CC(C(=O)NC1(CSC)CCC1)NC(=O)COc1ccn(C)n1 C(C)(CCCCNC(c1cncc(-c2cnn(C)c2)c1)=O)NC(C1C(C=C)C1)=O C1(NC(C2CCCC2)=O)CN(CCn2cc(CO)nn2)CC1c1ccccc1F c1(C(N2CCC3(C(NC(C(C)Cn4cncn4)=O)C3)C2)=O)cccc2ncsc12 c1(C(=O)NCC=CCNC(C23CC(F)C2C3)=O)c(C(F)(F)F)nc2ccccn12 N1(C(c2cc(C)[nH]n2)=O)CCCCC(NC(c2n[nH]c(C3CC3)n2)=O)C1 N1(C(C=COCC)=O)CCC(C2CC2)(CNC(C23CCC(CC2)C3(C)C)=O)C1 C1(CC)CCCCCCN1C(=O)C(n1cnc(C#N)n1)C C1(N(C)C(c2cncn2C)=O)CCCN(C(c2nc(Br)cs2)=O)C1 O=C(CC(C(F)(F)F)NC(C1CCS1(=O)=O)=O)NCc1noc(C(N)=O)n1 c1(C(=O)NCC(CCCC)NC(=O)C#CC(C)C)nccc(OC)c1C N1(C(C(C(C)C)C)=O)CCC(CNC(c2ccn(CC3CC3)n2)=O)C(F)(F)CC1 C12(C(=O)NCCNC(C3CCC(N(C)C)CC3)=O)CC3CC(C(=O)N1)C2C3 c1(-c2ccc(OC)c(C)c2)c(C(=O)N(C)Cc2cc[nH]n2)nn2c1CCCC2 N1(C(=O)NC2CCC(CNC(c3ccc(F)c(O)c3)=O)CC2)CCS(=O)(=O)CC1 c1(C(N2CC(C)N(C(C3CC4CC3C4)=O)CCC2)=O)ccc2ncn(C)c2n1 C1(N(C(C(C)OCC)=O)C)CCCN(C(=O)CCSc2ccc(OCC)cc2)C1 CC1(C)CC(=O)NCCN1C(C1(CS(C)(=O)=O)CCC1)=O C1(C#N)(C(=O)NCC(=O)NC(C)C(O)C(F)F)CC12CCC2 c1(C(N2CCCC(C)(CO)C2)C(=O)NCCCC)ccc(Cl)c2c1CCC2 CN=c1nc(N2CCOC(SC)C2)[nH]c(=NC(C)c2n[nH]c(=N)s2)[nH]1 c1(C(=O)NCC(C)Nc2cc(OC(C)C)ncn2)coc2ccc(F)cc12 N1(C(CC(C)C2CC2)=O)CCCC(CCC2CCN(C(c3ccco3)=O)CC2)C1 CCCC(C)CC(=O)N(C)CC1CN(C(=O)C(c2ccccc2F)(F)F)CCO1 n1(CC(=O)NC2C3(CC(NC(C(CC)C(C)C)=O)C3)C2)ccc(=O)c([N+](=O)[O-])c1 CC1CCC(C)N1CC(=O)NCC1CC(C)N(C(c2cn(C)nn2)=O)C1 C1(NC(=O)Cn2cncn2)CN(C(=O)Cc2cnc(C3CC3)[nH]2)C2(CCCC2)C1 Cc1cc(NCC2CC(NC(C3CCC4CC4C3)=O)C2)n2nc(C)cc2n1 C(C(C)C#N)N(C(C)C(=O)N(CCSC)C(c1cccs1)=O)CCC C1(N(C(c2c(CC)nns2)=O)C)CCCC2CN(C(c3sccc3CC)=O)CC12 Cc1nccc(C(=O)NC2(CF)CCN(C(=O)C=Cc3cnc[nH]3)C2)n1 c1ccc(C2CCN(C(c3cccs3)c3cccs3)C2)cc1 CCC(C)C(CNC(C1CCCN1C(=O)CC1CC(O)C1(C)C)=O)CO C12(C(N3CC(C(C)(C)O)(CNC(CC=C)=O)C3)=O)CC(C1)Oc1ccccc12 N1(C(C(=O)NCC(c2ccc(Br)cc2)(C)C)=O)CCC2CCCNC2C1 C1(NC(c2c(C)noc2)=O)CN(C(c2ccc3nncn3c2)=O)C2CCCCC12 CC1C=C(C(=O)N(CCCNC(C2CCCOCC2)=O)C)CC1 C(=O)(CCC(C)C)NC(C1CCCN(Cc2nc(Br)cn2C)C1)CC C(C(=O)NC1CCCOC1)(C1=CCSC1)N(CCCC1CCC1)C C1(CNC(C23CC(C(C)(C)C)(C2)C3)=O)CCCN(C(C2CCCC2CF)=O)C1 C1(C)(NC(c2c(CC)[nH]cc2)=O)CCCN(C(=O)CCS(=O)(=O)N(C)C)C1 C1(O)(CNC(C(C)(c2ccccc2)SC)=O)CCN(C(c2ccc(C)n2C)=O)C1 C1(CNC(CC(C)c2ccco2)=O)CCC(CNC(C2CC(C)CCO2)=O)CC1 C1(C(N2CCN(CC(=O)NCC3CNC(=O)O3)CC2)=O)CCC(F)(F)CC1 Cc1cc(N2CCCC(N3CCOCC3)C2)nc(=NCc2cnc(C)[nH]c2=N)[nH]1 C(=O)(C1=CC2(CCOC2)C1)N(CCNC(C(CN(CC)CC)F)=O)CCOC C(=O)(C(C(C)(C)C)NC(=O)CC1(C)OCCO1)N(C)CC1CCCCC1 CC1(C)Cc2ccc(C(=O)NC3C4CN(C(C5(CO)CCC5)=O)CC34)c(O)c2O1 C(=O)(CC(C)C(C)(C)NC(C1CC(N=[N+]=[N-])C1)=O)NC(C)CC1CCCCC1 N1(C(C2C(C)C2)=O)CCCC(C)(CNC(c2ccc(-c3cnn(C)c3)o2)=O)C1 c1(CC(=O)NCCNC(=O)C2=CCCC2)ccc(-n2ccnc2)cc1 n1(CC)ncc2cc(NC(=O)Nc3cnn4ccccc34)ccc12 S(=O)(=O)(c1cccs1)NC(C)C(N1CCC2C(NC(=O)CN(C)C3CC3)CC12)=O C(CC(C(=O)N(C)CC1(F)CCCC1)NC(=O)C(F)C1CCCC1)OCC C(C)(CNC(=O)C(C(C)C)N1CCCC1=O)(CC(C)C)NC(CSCC=C)=O C1(O)(C(C)NC(=O)CCCN(C)C)CCN(C(c2ccn(CC#N)n2)=O)C1 c1(C(=O)NCC(C)N(C(=O)C=Cc2cscn2)C)cc(Cl)c(Cl)n1C c1(CNC(C2C=COC2)=O)cccc(OCS(C)(=O)=O)c1.C12(CC1)C(=O)NC2 C=CC(C)(CC)C(=O)NCCCC1CCCN1C(=O)C(c1cc(F)ccc1F)=O CCC(CNC(c1ccc(NC(=O)NC)cc1)=O)N=c1[nH]c(Cl)c(C#N)s1 c1(C(=O)NC2CN(C(CC(C=C)C)=O)CC23CCC3)cc2cccnc2cc1F N1(C(CC(CC)(C)C)=O)CC2CC(NC(=O)CC3(O)CCOC3)C(C2)C1 C(=O)(C1=Cc2ccccc2C1)NC1CC2N(C(C3C(=C)C3)=O)C(CCC2)C1 c1(C(=O)NC2C(CNC(c3ccc(Cn4cccn4)o3)=O)C2)ncccc1F c1(C(N2CC3(C2)CN(c2ccc4nncn4n2)C3)C)sc2ccccc2c1C CC(C)C(O)C(C)C(=O)NC(C1CN(C(c2c[nH]nc2-c2cnn(C)c2)=O)C1)C C1(C2CCN(C(=O)C=C(CC)CC)CC2)(NC(C(CC)OCC)=O)CC1 N1(C(C(N2CCOCC2)C)=O)CC(=O)CC1C(=O)Nc1ccc(O)cc1 N1(C(C(C=CCCC)O)=O)CCC(CNC(=O)CCc2cccnc2F)(OC)C1 C1(C(N2CCCC(CC)C2)=O)CCN(C(=O)C(C2CCCCC2)=O)C(C)C1 CC1CCC(C)N1C(C)C(=O)NCCN(C(c1ccc(C(F)F)s1)=O)C1CC1 N1(C(C(C)NC(=O)OC)=O)CCCCC(CNC(c2coc(Br)c2)=O)C1 C(=O)(C(CCNC(=O)C=CCN1CCC1)OC)N(CC(C)(C)O)CCC c1(COC)ncc(C(N2CC3CC2C3NC(C23CC4CC2C3C4)=O)=O)c(=N)[nH]1 C1(N(C)C(C2(C)CCC(=O)C2)=O)CC2CCC(C1)N2C(C1CC1c1ccco1)=O c1(CC)conc1C(=O)NC12CC(NC(C3CCC(N(C)C)C3)=O)(C1)C2 C1(C)C(O)CO1.c1(NC(C(=O)NCC2(CCC)CCC2)=O)ccncc1 n1(CC(N2CCN(C(=O)CCN3CCC3)CC2)=O)ncc2cc(Br)cnc12 c1(C(=O)NCC(C)NC(C2CCC(C)(C)O2)=O)cc(Cl)ncc1N C1(C(=O)NCCCC(=C)C)C(C2CC2)CCN1C(c1cn(C)c(C)n1)=O N1(C(c2c(C)nc(O)cc2)=O)CC2CC(NC(C3(Cl)CC3)=O)C(C2)C1 N1(C(c2cn(C=C)nc2)C(=O)NCCOC(F)F)CCC(CO)(OC)CC1 c1(OC)ccc(Cl)cc1CC(N1CC(CNC(=O)CSc2ccccc2C)C1)=O N1(C(CNC(CC)=O)=O)CC2CCC1C1CN(Cc3ncnn3C)CC21 c1(C(=O)NC(CC)CNC(C2(Cc3ccc(O)cc3)CC2)=O)cc2cn[nH]c2cn1 C1(OC)CN(C(=O)CN2CCCS2(=O)=O)CC1NC(c1ccc(CCO)cc1)=O Cc1[nH]c(CCC#N)c(C)c1C(N1CCOCC1CNC(=O)C(F)C(F)(F)F)=O N1(C(CCc2cc(C)[nH]n2)=O)CCC(O)(C(C)NC(c2ncccn2)=O)CC1 c1(C(C)NC(c2ncoc2CNC(C2CC2(F)Cl)=O)=O)ccccc1O C(=O)(C(CCSC)NC(=O)C(C)=CCC)N(CC#C)CCF C(=O)(C1COc2ccccc21)NC1CN(C(CC2C(C)C(=O)CC2)=O)C2C1CCC2 C=C(Cl)CC(C(=O)N1CCCNC(=O)C1)NC(=O)CN1CCCCC1C Cc1[nH]c(C(N2CC(NC(=O)CC3CCC(C)CC3)CCC2C)=O)c(C)c1C Cc1cccc(Oc2ccccc2C(=O)NC2CC3CC2CO3)c1 N1(C(C23CC(C#N)(C2)C3)=O)CCC2CC2(C(=O)NC2CN3CCC2CC3)CC1 C1(CNC(C(C)Cn2ccnc2)=O)CN(C(c2ccnn(C)c2=O)=O)C(C)(C)C1 c1(C(=O)NC2CC(CCNC(C3(C(N)=O)CC3)=O)C2)cn(CC(N)=O)nn1 C(=O)(CCCC(=O)NCCN(C(C1SC2C=CC1C2)=O)CC1CC1)N(C)C N1(C(CC(C)CNC(=O)C(C)(C)C)=O)CC2(CCOCC2)C1 c1(C(N(CCCCNC(C(CC)=CCCC)=O)C)=O)cnc(OCC)c(C)c1 c1(CNC(=O)C(=O)N2CCC2C2CCC2)ccccc1N1CCOCC1 C1(C#C)(NC(C(C)(CO)NC(CC2CC(CC)C2)=O)=O)CC2CCCC12 c1(CC2C(C(=O)NCCNC(C(CN(C)C)O)=O)C2)cccc2ccoc12 C1(C2C(C(=O)NC3C(CCC(=O)NCC(C4CCC4)OC)C3)C2)CC(C)(C)C1 C1(NC(c2n(C)c(Cl)nc2)=O)CN(C(C2(CF)CCC2)=O)CC2(CCC2)C1 C(c1ccccc1C#N)=CC(=O)NC1(CNC(CC2CCC(C)CC2)=O)CCC1 O=C(N=c1cnn(C2CCOCC2)[nH]1)C1CCOC(c2ccccc2)C1 c1(C(C)C)cnn(C)c1C(N1CCC(C)(CNC(=O)C(C)CC2CC2)C1)=O n1(C(C)C)nccc1C1OCCC1C(N1CCC1NCC1CCCC1O)=O c1(OC)ccc(C(F)(F)F)c(C(N)=O)c1.N12CCC(CC1)C(=O)N1C(CC1)C2=O C1(OC)CN(C(=O)CCn2cncn2)CC1C(=O)NC(C)CCC1CC1 N1(C(C(n2ncc(C)c2)C)=O)CCC2(CC1)CC(NC(=O)C#CC1(C)CC1)CO2 c1(OC)ccc(C(F)F)cc1C(=O)NC(C)CCNC(=O)C=C(C)C(F)F CC(C)C(CCNC(c1cc[n+]([O-])cc1)=O)NC(c1cocc1Br)=O Cc1cccc(CC(=O)NCC2CCN2C(c2cccc(CCC(N)=O)c2)=O)n1 c1(C(N2CC(CC)N(C(=O)CC(C)(C)CC)CC2)=O)cn2c(n1)COCC2 N(C1CCCn2ccnc21)C(C(CC#CC)NC(c1coc(C2CC2)n1)=O)=O C1(NC(c2n3cc(C)sc3nc2)=O)CN(C(C2CCC(=O)O2)=O)CC1S(C)(=O)=O CN1CC2(CCN2C(=O)CC2CN(C(C3CCCOC3)=O)CCO2)C1 C(=O)(C(=O)CCC(C)C)NCC(CC(=O)NC(CC)CC)O Cc1cccc(C)c1OCC(N1CC2CC2(NC(=O)C=CC(F)(F)F)C1)=O C12(C(N3CCN(C(C(C)OC)=O)CC3C)=O)CC3CC(C(=O)N1)C2C3 N1(n2cc(CC#CC(=O)O)nn2)CC2C(CCO)C2C1 N1(C(=O)C=C2CCOCC2)CCCCC1C1CCCN1C(=O)Cc1cn[nH]c1 C(=O)(C(O)CC(F)(F)F)NCCCN(C(C1CCN(C)C(=O)C1)=O)C1CC1 N1(C(C(C)C2CCC2)=O)CC(C(=O)O)OCC12CCC2 N1(C(C(C)NC(C)=O)=O)CCC(F)C(NC(c2c(Br)sc(C)c2C)=O)C1 C1(CNC(C2C(C)C2C)=O)CCCN(C(=O)COc2ccc(Cl)c(F)c2)CC1 CC(C)CCC(O)C(=O)N1CCCCC1CC(=O)N(C)CC1CC1 CC(C(=O)NCC1CC(Nc2nc(C(C)(C)C)ns2)C1)C(F)F c1(CC)onc(C)c1C(=O)N(C1CC1)Cc1cn(CCC2CC2(Cl)Cl)nn1 CC(C)(CC(=O)N1CCCC12CCN(C(C13CCCC1C3(F)F)=O)C2)CC(F)F Cc1ccc([N+](=O)[O-])c(N2CCN(C(C3CCC=CCCC3)=O)CC(O)C2)c1 c1(SCCCC)ccc(CN(C(c2cccnc2S)=O)CC2CCOC2)cc1 C(C(O)CN(C)OC)NC(C(CC)Oc1ccccc1F)=O N1(C(C(C(C)C)NC(C(CNC(C)=O)(C)C)=O)=O)CCOC2(CCC2)C1 c1(C(N2C(C(=O)Nc3ccnnc3)CCC2)=O)cnc2ccccn12 c1(OC)ccc(C(=O)NC2(C3CCCCN3C(c3cnns3)=O)CC2)cc1 N(C(=NCCCOC(C)C)NCc1cc(C)nc(C)c1)CC(C=C)C c1(C(=O)NCC2C(C)(C)CN(C(c3ccccc3)=O)C2)cc(F)c(N)c(F)c1 CC1(C)C(CC(=O)NCC2CC(NC(c3ccc(SC(N)=O)cc3)=O)C2)C1(C)C Cc1ccc(C)c(C(N2CCC(N(C(=O)CN3CC(=O)N(C)C3=O)C)C2)=O)c1 CC(CC1=CCCCC1)NC(C1COCCC1NC(=O)C=C1CCOCC1)=O c1(C2N(CC(CSC)OC)CCCC2)ccc(O)cc1 c1(NC(=O)NC(c2ccc(Cl)cc2)C(C)(C)C)cccc2nc(O)ccc12 N1(C(CC(C(F)F)OC(C)=O)=O)CCOC(C)(C)CC1.C12(CC1)C(=O)N2 C1(CCCNC(C2CCCC2C)=O)(CNC(C2(CCCC)CC2)=O)CCCC1 Cc1cc(C(C(=O)NCC2CC2)N(C)C(C2CCOC2)C)ccc1I.c1(C)ccsc1 N1(C(COc2cccc(C)c2)=O)CCN(C(=O)C2CC2)CC1C1CC1 C12(NC(=O)Nc3c(CN(CC)CC)c(CC)ccc3)CCC(CO)(CC1)CC2 CC(C(=O)NCC1CCC(F)(C(=O)NC)CC1)C(C)C(C)(C)C.C1(=O)C(=O)C1CC C1(NC(CC2ON=C(CC)C2)=O)(CNC(C2(C3(C)CC3)CC2)=O)CCCCCC1 O=C(C1=NOC2(CCOC2)C1)N1CCN(C(C23CCCC2C3(F)F)=O)CC(O)C1 Cc1cccc(C2CC(c3nnnn3C)(NC3(c4ncco4)CC3)C2)c1 c1(C(=O)OCC)[nH]cc(CNC(C)Cc2nn[nH]n2)c1C c1(C(=O)NCC(CC)NC(C2CCCCC2O)=O)coc(S(N)(=O)=O)c1 CCCC(C(=O)NCC1CC2(CC(NC(C3CCC3CF)=O)C2)C1)S(N)(=O)=O Cc1noc(C)c1CCc1nc(-c2ccn(C)n2)nn1CCN(C)C C(=O)(N=c1ccc2nccn2[nH]1)c1cc(C(=O)OC)n[nH]1 C1(C(=O)NCc2c(C)cccc2)CN(C(=O)C(F)CC2CCOC2)CC(C)(C)C1 c1(C(N(CCCN(C(=O)C(F)C2CCOC2)C)C)=O)cc(F)cc2nc(S)[nH]c12 c1(C(N(CCCNC(C2CSCC(=O)N2)=O)C(C)C)=O)cc2c(=O)[nH]ccn2c1 C(C1CCCN1C(=O)Cc1cn(C)cn1)=CC(=O)NCC1CCC(C(N)=O)O1 C(=O)(C(CNC(=O)CC1CC2C=CC1C2)CC=C)N1CCC(OC)C1C N1(C(CC2(C)CC2)=O)CC2CCCC1C2CNC(C1(C)CC1(F)Cl)=O N1(C(C23C(C)OC(CC2)C3)=O)CC2CCC(NC(=O)CSCC(F)(F)F)(C2)C1 C(CC(C)CCNC(c1cn(C2CC2)c(O)n1)=O)NC(c1cnc(C(C)C)[nH]1)=O N1(C(C(C2CCOCC2)OCC)=O)CC2C(CNC(=O)CCc3ccco3)C2C1 CC1(C)CCCN(c2cc(Cl)nc(CO)n2)C1CNC(C12CC1COC2(C)C)=O C1(CNC(C(CC)O)=O)CN(C(=O)C(c2cncnc2)C)CC1(F)F c1(OC)c(C(=O)NC(C)CC(C)NC(c2cc(C#N)cs2)=O)ccc(Cl)c1C c1(CCCN)cnn(CC(F)F)c1C.c1(COCC)nc(CNC(=O)OC(C)(C)C)no1 CC1(C)OCCC1CC(=O)NCC1(CO)CCN(C(C23CC(CO)(C2)C3)=O)C1 C(CCC)(C(=O)N1CCC(O)(CCNC(=O)COc2cc(C)on2)C1)=CCC C=CCC(C(=O)N1CCOCC1C(=O)NCC1CCCSC1)NC(C)=O S(=O)(=O)(c1ccc(NCCCOC2CCN(C)CC2)c(Cl)c1)NC(C(C)C)CCO c1(C(N2C(CNC(c3ccc(CC)o3)=O)CCC2)=O)cc(F)cc2nn(C)cc12 N1(C(CC(CC)SC)=O)CCCC2CN(C(C3(CC)CC3)=O)CCC12 N1(C(c2cc(C)nn2C)=O)CCC(F)(CNC(C2(C)CCCC2O)=O)CC1 Cc1cncc(C(=O)NC2CCN(C(c3ccc(C)n3C)=O)C(C3CC3)C2)c1Cl C1(OC)CN(C(=O)Cn2ccnn2)CC1NC(=O)Cn1cc(C2CCOC2)cn1 c1(C(=O)OC)cnn(C)c1C(=O)NC1CC1NC1(C(N2CCCC2)=O)CC1 N1(C(C(CC)n2ccnc2)=O)CCCC(CCNC(C2(F)CC2)=O)C1 c1(C(=O)NC(CC(C)NC(C=CCOC)=O)C)ccn(CS(C)(=O)=O)n1 Cc1cc(N2CCC(NC(=O)CCCCN(C)C)C2)nc(CO)n1 c1(C(N2C(C)(CNC(c3cccc(C)c3F)=O)CCC2)=O)ccc(F)c(C)c1C c1(C(=O)NCC(C)(C)NC(C(C(C)SC)O)=O)ccc(Br)c(C)n1 CC1CN(C(=O)C(C)N(C(=O)C(c2ccn(C)n2)C)C)CC(CO)O1 C1(C(N2C(C)(CNC(c3cn(CCC=C)nn3)=O)CCC2)=O)C(F)(F)C12CCC2 C1(CCC(N2C(C(CC)C)CCC2)=O)CCCC2(CC2)C1 C(=O)(C1=C(C)CCOC1)NCC(CCCC)NC(c1csc(CCC)n1)=O CN1CC2CN(C(C3(CNC(C4COCOC4)=O)CCCC3)=O)CC2C1 C=Cc1cnn(C)c1C(=O)NCCC1(O)CN(C(C2CCCNS2(=O)=O)=O)C1 C1(C)(CNC(C2C(CC)CCC2)=O)CCN(C(=O)CC2C=NN(C)C2=O)C1 C1(O)(CC(C)C)CN(C(C2CCC2NCc2nc(N(C)C)co2)=O)C1.C(=O)OC N1(C(C2(CC=C)CCN(C(C3(C#N)CCOCC3)=O)C2)=O)CC2COC(=O)C2C1 N1(C(c2c(C)ocn2)=O)CC(CNC(=O)CN2CCOC2=O)OC2CCCC12 C1(NC(c2c(CC)nc(C)[nH]2)=O)C2CC1N(C(c1ncc(Cl)cc1F)=O)C2C C(c1c(C)nn(C)c1Cl)=CC(=O)NCC(CO)NC(Cc1ccc(C)nc1O)=O C(=O)(CC(CC)C(C)C)NCC1(O)CCN(C(c2cncc(C#C)c2)=O)CC1 c1(C(N2C(C(=O)NCCSCC)CC3CC32)=O)ccc2nc[nH]c2c1 CCCCC(C)N=c1[nH]c2c(c(=NCCC(C(C)C)NC(=O)NC)[nH]1)CCC2 c1(CCN2CC2=O)ccccc1.C1(CN(C2(C)CCC2)C2CC2)CC=CCC1 C1(NC(C(=O)NCC2CC3C4C=CC(C4)C23)=O)CCCN(C2CCC2)C1=O c1(NC(C2C(NC(c3ccn(C)n3)=O)CC2)=O)ccc2cnn(C)c2c1 c1(CCN(CCC(=O)NC(=O)NC2CCOC2)CC)ncoc1C c1(CCCC(=O)N(CC(CNC(C(C)CF)=O)(C)C)C)c[nH]c2ccccc12 C#Cc1cccc(NCC2CCCC(N)C2)c1.N12CCCC(CC1)NC(=O)C2 N1(C(CCNC(=O)NC)=O)CCC(C2CC2)C1C(=O)Nc1ccc(OC)cc1 C=CC(CC)CC(=O)N1CC2CC1CN2C(C1CC2(C1)CC2F)=O Cc1cc(C(=O)NC2CCCCC2N(C)C(c2cn(C3CC3)nn2)=O)cnn1 N1(C(C2(C#C)CN(C(=O)CSCC)C2)=O)CC2CC(C1)C2(C)C N1(C(C)C)CCOC(C(=O)NC(C)CNC(c2c(C(C)C)cnn2C)=O)C1 C1(C(=O)NCC(C2CCC2)OC)CCN(C(=O)c2ccc(C)nc2)O1 N1(C(C2(C)CC=CC2)=O)CCC(C)(CNC(=O)Cn2cnnn2)C1 c1(OCC)c(OC)cc(C(N2CC(N3CC(NC(=O)CC)CC3=O)C2)=O)cc1Cl n1(CC)nc(-c2ccc(SC3(C)CC3)cc2)nc1C(N1CCOCC1)C(C)C N1(C(C)C)CCN(CCC(=O)NCC(=O)CC2CCOC2)CC1 N1(C(C2ON=C(C)C2C)=O)CCC2(CC1)CN(C(=O)CC(C)n1cccn1)C2 N1(C(CCOCCOC)=O)CC(F)CC1C(=O)NCC(C1CC1)C1CC1 c1(C(=O)NCc2occ(C(=O)NCC(=C)CC)c2)ccc2cncn2c1 C1(C(N(CCC(=O)NCc2ccc(CC)s2)C)=O)CCC(C)(O)CC1 c1(CNC(C(C2CCC2)OCC)=O)ccc(C(=O)NCCCN=[N+]=[N-])nc1 c1(C(N(CCCCNC(CCOCC(C)C)=O)C)=O)ccc(O)nc1 c1(C(N2CCC(OCC(C)C)C2)=O)coc(C(C)NC(C2CC3(CC3)C2)=O)n1 c1(C(N2CC(C)C(NC(c3cc(F)cc(F)c3)=O)C2)=O)ccc2ncncc2c1 c1(N(C(=O)C(C)(C)Br)C(C2CCCNC2)C)nc(Cl)c2c(ccn2C)n1 N1(C(c2c(C)cncc2)=O)CCC(NC(=O)CC2(C)OCCO2)C(C)C1 C#CC1(O)CCN(C(C2CCN(C(c3cnc(CC)o3)=O)C2C)=O)C1 c1(C(C(=O)NCc2ccco2)N(C(CCC)C)C)ccc2c(c1)CCC2 CCC(CC(F)(F)F)NC(C1CC(CNC(c2ncn(CC)n2)=O)C1)=O C1(CNC(=O)CCc2ccon2)CCCCC1NC(=O)CC1CCC1 c1(CC)c(C(=O)N(CCNC(C2CC2F)=O)CC2CC2)oc2ccc(Br)cc12 N1(C(C2(SC)CCC2)=O)CCC(CNC(=O)CCC2CCCO2)C(O)C1 C(=O)(C1=C(C)CCOC1)NCC(C)CC(=O)N1CCCC(CO)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N(CCOCCN(C(=O)CN1CC=CC1)C)C CC1(CNC(C2CC2F)=O)CCCN1C(c1nc(Cl)c(Cl)s1)=O C(=O)(C1=NOC(CNC(C2CN(C(N)=O)C2)=O)C1)NCC1(C)N=C(C)SC1 N1(C(C2C(C(=O)OC)CCO2)=O)CCC(NC(=O)CCCC(N)=O)C(CO)C1 C1(CCNC(C2(CCCC)CC2)=O)C(C)CCCN1C(c1cnc(C(C)C)s1)=O C1(NC(C=CCN(CC(F)(F)F)C)=O)CC2(CCCN(C(C3CC3(F)F)=O)C2)C1 C1(CCNC(=O)OCc2cccnc2)(OC)CCC1 Cc1ccc(NC(C2CCN(C(c3cnsn3)=O)CC2O)=O)c(Br)n1 C1(CNC(=O)CC2CC2C2CC2)CC(O)CN1C(=O)CCC(=O)c1cccs1 CC1CCc2c(Cl)cccc2C1NC1CC(CC(=O)O)C1(C)C C12(C(N3CC(NC(C(=O)NCCC(N)=O)=O)C3)=O)CCC(C(F)F)(CC1)C2 c1(OCC)nc(N2CCCC2CC(=O)NC2CCCN(C)C2)ncc1Cl c1(C(=O)NCCCN(C(C2C(C)(CC)C2)=O)C)c(O)cnc2ccccc12 N1(C(C(C=CC)O)=O)CCOC(C)(CNC(=O)Cn2nc(C)c(Br)c2C)C1 c1(CNC(=O)C(N2CCc3ncsc3C2)=O)ccc2c(Cl)csc2c1 CC(CN=C(NCC(F)F)NCC(c1ccccc1)CO)S(C)(=O)=O Cc1nc2c(o1)CCCC2CC(=O)NC(C)CCCNC(C1CC1F)=O N1(C(C=CC(C)=O)=O)CCC(C)C(CNC(c2ncccc2C2CC2)=O)C1 C1(C(=O)NC2CCC(CCC(=O)NCc3c(C)ccnc3)C2)CC(C)CC(=O)N1 C12(CNC(c3c(N)non3)=O)CN(C(=O)Cc3ccccc3)CC1CS(=O)(=O)C2 c1(OC)ccc(NC(=O)C(C)NC(C2CCC2C)C)c(OC)c1 CCCCCC(C)CC(=O)N(C(C)(C)CC(=O)N(C(C)CCC)C)C C1(C(=O)NCC(CC=C)NC(c2cccc(F)c2)=O)CC(F)CN1C c1(NC(=O)NC(CC=C)C(=O)OC)nc(OCCC)cc(C)n1 C(C1=CCN(C(=O)CNc2cc(Cl)cc(Cl)c2)CC1)NC(c1c(CC)csc1)=O c1(OCC)c(C(=O)N(C)CC2(CNC(=O)CCCSC)CC2)cccc1F C1(COC)CN(C(C2CC=CCC2)=O)CCN1C(=O)COCc1cc(C)on1 c1(C(N(CC(CN(C(c2ccc(C#C)o2)=O)C)O)C)=O)cc2nc[nH]c2cc1N c1(N(C(C)C)C)ccc(C(=O)N(C)Cc2cccc(F)c2)cc1[N+](=O)[O-] c1(C(N2CCC(C)C2CNC(c2nn(C)cc2Cl)=O)=O)ccc(F)c(C#N)c1 N1(C(CC(CC)C2CC2)=O)CC2C3CCC(C2C1)N(C(c1nnccc1C)=O)C3 N1(C(CCCOCC)=O)CCC2CCN(C(c3cc(Br)co3)=O)CC12 N#Cc1ccc2c(c1)CCN(C(C1CN(C(c3ccnc(F)c3F)=O)CCN1)=O)C2 c1(OCC(=O)NCC(C)NC(Cc2cc(C)[nH]n2)=O)ccc(Br)c(C)c1 N1(C(c2ccn(C(F)F)n2)=O)CCCC(O)(CNC(C2(CF)CC2(F)F)=O)C1 CCCC(CCCNC(=O)C(C)NC=O)NC(=O)Cn1cnnn1 C1(CC=C)(C(=O)NC(C2CCCC2)CNC(c2coc(OC)n2)=O)CCOC1 C(=O)(CS(=O)(=O)NC1CC1)NCC(CN(C(=O)CCn1cncn1)C)(C)C CN=C(NCCC1CCCO1)N1CCC(C(N2CCC2c2ccccc2)=O)C1 S(=O)(=O)(CC(=O)NC1CN(C(=O)C=CC2CCCCC2)CC1C)NC CC1(NC(=O)CC2CCC(C)(C)CO2)CCCN(C(=O)C2=CCCC2)C1 C1(C(N(C2CCN(C(c3sc(CC)c(C)c3)=O)C2)CC)=O)Cc2cccnc2C1 C1(NC(=O)C=C2CCCCC2)CC2CC1CN(C(=O)Cc1cccc(Cl)c1Cl)C2 CC1(O)CCC(C(=O)NCC(O)CNC(=O)CC2CC(F)C2)CC1 CC(C)(CC(=O)N1CCCC1CNC(C1CCS1(=O)=O)=O)CCCc1nccs1 c1(CC(=O)NC2(CCCNC(COC)=O)CC2)c(F)cncc1Cl c1(CC)ncc(C(=O)NCC(C)N(CC(=O)N(CC(C)C)CCOC)C)o1 c1(C(=O)NCc2scc(C(C)NC(=O)NC(C)(C)C)n2)cc(I)ccc1[N+](=O)[O-] CC1CCC(NC(=O)C(C)(C)C)CN1C(c1cnn(CC2CCC2)c1)=O N1(C(c2cc(C)c(Cl)s2)=O)CCC2(C1)CN(C(=O)C(N1CCSCC1)C)C2 c1(OC)nccc(N2CC3C(C(=O)NC(C#N)C(N)=O)C3C2)n1 N1(C(C2N(C)CCCC2)=O)CCC(NC(=O)CCC2CCOC2)C(C)(C)C1 CC1CC(C)N(C(=O)OCCOC(C)(C)C)c2ccccc21.C1(=O)C(C)(CO)O1 N1(C(c2cnc(C(N)=O)s2)=O)CCC(NC(=O)CC2COC3CC2C3)CC(O)C1 c1(C(N(CCCNC(=O)CSCCC#N)CC)=O)cc(C#N)no1 CCS(=O)(=O)CC(=O)NC1CCN(C(c2cn(C(C)C)nn2)=O)C1C1CC1 C(C(COC)C(C)C)NC(C(CC)C)=O.C12(CSC1)C(=O)N2 c1(NC(c2scc(C(=O)Nc3cccc(CC)n3)n2)=O)ccc(Br)nc1Cl C1(C(N(C)CC2(CNC(=O)C3=CCCCC3)CC2)=O)CCC2(CCOCC2)C1 C(C)(C)(C(=O)NC(C)CC(C)NC(=O)Cc1csc(C)n1)OC c1(OC)cc(Br)c(F)cc1NCC1CC12CC2(F)F C1(NC(c2cc(CC)on2)=O)CCCC12CN(c1nnc(C(F)(F)F)s1)C2 c1(C(C)C)nc(NCCN2CCOC3(CCC3)C2)cc(=NC2CCCC2C#N)[nH]1 CCCCC(F)C(=O)N1CC(NC(c2cc(C3CCOCC3)nn2C)=O)C1 CN1CC(C)(C)CC1C(=O)NCCCCCNC(C1(C)CNC(=O)C1)=O N1(C(CCCCCNC(C)=O)=O)CCC2CCN(C(=O)C=Cc3cc[nH]n3)C2C1 C1(C(=O)NC(c2cn(C3CCCC3)nn2)C)Cc2ccccc2CN1 c1(OC)ccc2c(c1)OCC(C(=O)NC1CCC1CNC(c1c[nH]cc1C)=O)=C2 c1(C(=O)NC2C3CN(C(c4ccc(CC)s4)=O)C2C3)cc2cccnn2c1 c1(CC(N2C(CC3N(C(C)=O)CCC3)CCC2)=O)ccc(Cl)c(C)c1 N1(C(c2c(C(C)C)ocn2)=O)CC2(CCC(CNC(C3CC3C(C)O)=O)O2)C1 N1(C(C(c2cn(C)nc2)NC(c2csc(S)n2)=O)=O)CCC(C2CCCC2)C1 c1(CNC(c2cnn(-n3cc(-c4cccs4)nn3)c2)=O)ccoc1C1CC1 C1(CCNCc2cccc(C(F)(F)F)c2)Cc2ccccc2C1 Cc1cc(C(N2CCCC(CCNC(C3CC(O)C3)=O)C2)=O)ncc1Cl n1(C(C)C(=O)NCC(=O)NCC2CC2)cc(C2CCN(C)C2)nn1 C1(C2CN(C(=O)C3CC3)C2)(NC(C2CC2(F)Br)=O)CC1 c1(OC)cccc(C(C)(CC(=O)O)NC(=O)Cn2cc(C(C)(C)C(C)C)nn2)n1 c1(OCC(=O)NC(C2CCN(C(Cc3nc(C)oc3)=O)C2)C)ccc(C)c(C)c1 C1(C(N2CC(CC(CNC(CCCCC)=O)(C)C)C2)=O)CC2(CCO1)CC2 C1(CNC(C=CC(C)(C)SC)=O)CCOC1CNC(=O)CCC=CC(C)C C(C(C)(C)C(=O)NCC1CC(NC(c2cccnc2Cl)=O)C1)SC C=CC(CCC)CC(=O)NCCCCNC(=O)CC1CCS(=O)(=O)C1 c1(C(N(CCNC(C2C(C=C)C2)=O)CCC)=O)cc(N)ccc1Br CN1CCCC1C=CC(=O)NC(CCOCCO)C(=O)Nc1cnn(CCO)c1 c1(SC)nc(N2CCN(C(c3cc(-c4ccco4)no3)=O)CC2CO)ncc1F C(C#Cc1ccc(F)cc1)N1C(CCNC(c2cc(OC)n[nH]2)=O)CCC1 c1(CC(=O)N(CCN(C(C(CCNC(C)=O)C)=O)C(C)C)C)c(F)cncc1Cl C12(CNC(c3cc(OCC)n[nH]3)=O)CC1CN(C(=O)CCC(=O)N(C)C)C2 c1(C(CCN(C(=O)C(=O)NCc2cnsc2)C)O)ccccc1 N1(C(C2(NC(C)=O)CCCC2)=O)CCC2CN(Cc3ccc(Cl)cc3F)CC12 S(=O)(=O)(c1cnc(N(C2(C#N)CCC2)C)cc1C)N(CC(CCC)O)C N1(C(CCN(CCC(C)(C)C)C)=O)CCC(C)(NC(=O)C(O)c2ccco2)C1 C1(CC(=O)NC2(CNC(=O)CCOC3COC3)CCCC2)CCCC12CC2 N1(C(C(C2CCOCC2)OC)=O)CCC(O)(CNC(c2nocc2Br)=O)CC1 N(C(=NCCF)N1CCC(CN2CCCCCC2)C1)C(C#C)C(C)(C)C C1(C(=O)NCC2CC(F)(F)CN2c2ncnc(Cl)c2Br)CCc2nnnn2C1 O=C1NCCCCC1CC(N1CC(OCCC(=O)N2CC(c3ccn[nH]3)C2)C1)=O N1(C(C=CC)=O)CC2(C1)SCCC2NC(=O)C(CC(C)(C)C)c1ccc(Cl)cc1 N1(c2n(CC(=O)N(C)C)ncc2)CC2CCCCCCC12 C#CCCCCC(=O)NCC1CCC1NC(=O)CCc1c(F)cccc1Cl C1(CNC(C=CC)=O)CCCN1C(C)=O.C12CCN1C(=O)C2 c1(C(N2CCOC(CCNC(C3(CCF)CCOCC3)=O)C2)=O)ncccc1O C1(NC(C(=O)NC(C)C)=O)CCCC12CN(C(C13COCC1C3(F)F)=O)C2 C1(CNC(C(F)SCC)=O)CCN(C(c2ccc(N3CCC3)cc2)=O)C1(C)C CC(O)C(C(=O)OCCNOCCO)N(C)C.C1CC(=O)C(=O)N1 C1(NC(c2cc(C)c(F)cn2)=O)CN(C(c2nn(C)cc2N)=O)CC(F)(F)C1 Cn1cc(S(N)(=O)=O)cc1CC(=O)NC1CCCN(C(=O)COC2CCOC2)C1 C=CCC(CC)C(=O)N1CCC(CCC(N2CCN(C)C(=O)C2)=O)CC1 CC1(C(N2CCC(C(F)F)C2)=O)CCN(C(=O)C=Cc2ccncn2)C1 C1(OC)(OC)CCN(C(=O)Cc2ccc(F)cc2C(F)(F)F)CC1 CC1(NC(c2cnco2)=O)CCCN(C(C2CC3CC3C2)=O)C1 c1(OC)ccc(CNC(=O)NCC2CCCC(C3CC3)O2)cc1Cl C=CCCCCCC(=O)C(C(CO)N)=O.C(C)(C)(C(O)CO)N CCCCC(CNC(=O)C(C)(C)c1ccncc1)NC(=O)C=CC(C)C C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC(C1CCN(C(CC(=C=C)C)=O)C1)C c1(N(C2CNCCOC2)C(C2CCC(C)O2)=O)ncnc2c1c(Br)cn2C c1(CC(=O)OC(C)C(=O)NCc2ccc(-n3cccn3)cc2)ccc(Br)cn1 C1(C(=O)NCCN(C(=O)CCc2cccc(C)c2)CC)CCCOC1C n1(CCC=C)cc(C(=O)NCC2CCCC2NC(=O)COCP(C)(C)=O)nn1 c1(C(N2CC(C3C(C(N4CCC(C(=O)NC)C4)=O)C3)C2)=O)ccn2cncc2c1 C(=O)(C(C)N=c1cc[nH]cc1)NC(CCNC(CCN(CC)CC)=O)(C)C C12CC3CCCC3N1C(=O)CCOC2=O.Cc1nnc(NC(=O)C(C)(C)C)s1 C1(C2CN(C(c3cnc(C)nc3)=O)C2)(NC(CCNC(=O)NC)=O)CC1 c1(CC(=O)NCCCCC(C)NC(C2C(C)C2(F)F)=O)ccc(S(C)(=O)=O)cc1 N1(C(c2cc(C)n(C3CC3)n2)=O)CC2CCC1CN(C(c1cn(C)cn1)=O)C2 N1(C(CCC(C)N(C)C)=O)C2CCC1CN(C(c1cccc(=O)o1)=O)C2 Cc1ccc(CN(CCO)C(C2C3CC2N(C(=O)Cc2sccc2C)C3)=O)nc1 C1(CNC(c2[nH]cc(C#N)c2)=O)CC12CCN(C(=O)CCCN1CCCC1)CC2 C1(C(=O)NCc2cnccn2)CCC2CCCCN12 N1(C(C(C(C)C)NC(C(CC)OC)=O)=O)CCN(C(C)C)C(=O)C1 C1(NC(C(C)O)=O)CCN(C(C2CC23CNC3)=O)CC1 n1(CCOCC)nnnc1C(c1cccs1)NCC1(C(C)C)CC1 c1(C(=O)NC(C(N2C(CCC)COCC2)=O)CC2CCC2)cc2ncccc2[nH]1 c1(C(=O)Nc2nnc(CC(=O)NCC)s2)cc(O)ccc1OC(C)C Cc1cnc(C(=O)N(CCC(C(C)C)NC(C2(F)CC=CCC2)=O)C)c(F)c1 c1(C(N(CC(C)NC(C(C)SCCCC)=O)CC)=O)cc(Cl)no1 N1(C(C2(OC)CC2)=O)CC2=C(C1)CN(C(C1(C)CCC3CC3C1)=O)C2 N1(C(c2nc(CC)sc2)=O)CCC2CN(C(c3ccn(C(C)C)c3C)=O)CC12 C1(NC(CCCC2C(C)C2)=O)(COC)CCCN(C(=O)C(=O)NC2CCCC2)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CCC2C(C1)CN2C(c1nccnc1N)=O Cc1ccc(O)c(CC(=O)NC2CN(C(=O)CCC34CCC(CC3)C4)CC2C)c1 N1(C(Cc2nc(C)sc2)=O)CC2CC(C1)CN(C(=O)CCC1(C)CC1(F)F)C2 CCCC(C)CCNCC(=O)NCC1CC1 c1(SC)ccc(NC(N2CCN(C(=O)C(C)Sc3ccccc3)CC2)=O)c(F)c1 C(=O)(CC1OCc2ccccc21)NC(CCOC)C(C)C C1(C(NOCCCC)=O)(NC(c2n[nH]cc2Cl)=O)CCCC1C c1(NCC(=O)N(C2CCC(NC(=O)C(C)(C)C)C2)C)ccccc1Cl C1(C(=O)NCC2(C)N=C(C)SC2)CCC(CNC(C2(NC(N)=O)CC2)=O)CC1 Cc1cc(CC(=O)NCc2ncoc2CCNC(=O)C(Cl)=CCl)cc(O)n1 c1(OC)cc2ccc(C(=O)NCC(F)CNC(c3ccccc3)=O)nc2cc1F N#Cc1cc(C(=O)NCc2cc(C(=O)NCCCc3ccco3)on2)cs1 N1(C(c2c(C)cccc2)C(=O)NC2COC2)CC(=O)N2CCCCC2C1 C1(C(=O)NCCC2CN(C(c3ccc([N+](=O)[O-])s3)=O)C2)CCc2ccccc2O1 c1(C(N2CCC(CN(C(C(CC)(CC)CO)=O)C)C2)=O)csc2cc(Cl)cnc12 O=C1CC(C(N2CC=CC(NC(=O)CN3CCCCCC3)C2)=O)NC(=O)N1 c1(SC)ccc(NC(N2CCCN(C(C)=O)CC2)=O)cc1Cl C(C(CC(C)C)NC(c1nc(C(C)C)oc1C)=O)NC(C(n1ncc(C)c1)C)=O C1(C(=O)NC2(C(=O)NCC(CC=C)(F)F)CCSC2)CN2CCC1CC2 CC1CN(C(=O)C(O)Cc2ccccc2)CCC1NC(c1ccc(NC)cc1)=O N1(C(C(CCC)O)=O)CCN(C(=O)Cc2ccc(OC)c(F)c2)C(C)C1 c1(C(N2CC3C(NC(c4ccn(CC)c(=O)c4)=O)C3C2)=O)ccc(C#N)nc1O c1(C(C2CC2)NC2C(C(C)C)CN(C(=O)C(C)N(C)C)C2)ccc([N+](=O)[O-])cn1 CCC(C)C(O)CC(=O)N1CC(C(O)C(N2CCCN(C(=O)OC)CC2C)=O)C1 C1(CC(=O)Nc2ccc(O)c(CO)c2)CN(C(=O)CC2CC(F)(F)C2)CC12CC2 c1(N2CCC(C(=O)OC)(CC)C2)nc(=NC2CC(CO)C2)[nH]c2c1CSC2 C1(N(C)C)CN(C(C2(CF)CCN(C(C3CCCN3C)=O)C2)=O)CC12CC2 c1(CNC(N(C)CCOC)=NCc2ccc(OC)cc2)nnc2ccc(C)nn12 C(C)(C)(C(=O)NCCCN(C)C(c1cc[nH]c1C1CCC1)=O)OC(C)C c1(CCC)[nH]nc(C(N2CCC(O)C(NC(=O)C3=CCCC3C)C2)=O)c1[N+](=O)[O-] N1(C(c2[nH]c(=N)sc2)=O)CCCCC(CNC(=O)CCCCCF)C1 C(=O)(CC(C(C)C)NC(c1cc(OC)ncn1)=O)N(CC=C)CCC CC1CCN(C(C2C(C)(C)OC2(C)C)=O)CCN1C(=O)CCCc1ccccc1 C1(OC)CN(N2CCCCC2CCC(C)C)CC(C)(C)C1 c1(OC)ccc2nc(NC3CC3C(F)(F)F)[nH]c(=NCC(CO)OC)c2c1 C(=O)(CC(C)C(F)(F)F)NC(CC#CC)C(=O)NCC1(C)CCC(=O)N1 C1(NC(C2(C)CC=CC2)=O)CCC2CCN(C(=O)CS(=O)(=O)C3CC3)C1C2 C1(NC(C(c2ccc(Br)cc2)C)=O)CC2CC1CN(C(=O)CCCF)C2 CCCC(C)CC(=O)N(C(C)CNC(=O)C(CC)n1cncn1)CC S(=O)(=O)(c1ccc(CBr)cc1)N1C(C(=O)Nc2cc(OC)nc(Cl)c2)CC(C)C1 O=C(C1=NN(CCO)C(=O)CC1)NC1CCCCC1NC(C1CC(F)(CO)C1)=O C1(CNC(c2cc3c[nH]cnc-3n2)=O)CCN(C(c2cccnn2)=O)C12CCC2 C1(NC(C#N)CC2CC2)CCC(C(=O)O)C1.n12cc(nn1)NC(=O)C2C C(C(=O)N1CCCO1)NC(C(CSCC)NC(C(C)SCCCC)=O)=O CC1(NC(=O)CCc2ncco2)CCN(C(c2c[nH]c(Br)c2)=O)CC1 c1(CC)nc(N(CCCNC(c2cc(OC)ns2)=O)CC)cc(C)n1 C(=O)(C(CN(C)C)CC)NCCC(CNC(c1nc(CC)oc1)=O)O c1(C(N(C)CC2N(C(CCOC)=O)CCOC2)=O)ccc2ncsc2c1 C(CCCC(CO)NC(=O)C(c1ccc(F)cc1)F)NC(C1(C(C)(C)OC)CC1)=O N1(CCC(=O)NCC2C(NC(C3(c4cccs4)CC3)=O)CC2)CCCCC1 CC(C)(C(=O)OC(C)(C)C)CCC(=O)NCCC1CCCCC1C(=O)O C1(C(C)C)CCCC1C(=O)OCc1ccc(C(N)=O)o1 N1(C(CCc2cn(-c3c(C(=O)O)cccc3)nn2)=O)CCCC2(CC2)C1 N1(C(c2c(C)nc(C(C)C)nc2)=O)CCCC2CCN(C(C3(C)CSC3)=O)CC12 c1(C(=O)NC(CC)CNC(c2c(OC)cccc2C)=O)cc2cc(C)ccc2[nH]1 c1(-c2ccc(C(=O)OCC3COC3)s2)cc2ccccc2s1 C(=O)(C(CC(C)C)C(N)=O)NC1CC2(CC(NC(Cc3cc(C)sc3C)=O)C2)C1 c1(C(N(CC(CC)NC(c2c(C)csc2Cl)=O)CC)=O)cccc2ncn(C)c12 C1(C(=O)NCc2cccc(=O)o2)CCN(C(=O)CCc2cccc(Br)c2)CC1 c1(C(=O)NCC2C(NC(C3CCN(C(C)=O)C3)=O)C2)ccc(N)c(F)c1 c1(C(N2CCC(CN(C(c3cnc(C)s3)=O)C)C2)=O)cc(O)nc2c1CCCC2 Cc1nc(C)c(C(=O)N(C2CC(NC(=O)C(F)(F)c3cncs3)C2)C)nc1C c1(C(C)N(C)C(c2cnc(Br)o2)=O)cccc(-n2ccnc2)c1 c1(C(=O)NC2CCC(C)(CNC(c3n(C)cnc3)=O)CC2)cc(F)cc(F)c1O CC1CN(C(=O)CCn2cccn2)CCC1C(=O)NC1CN(C(N)=O)C1 N1(C(c2c(C)nc(CNC(c3cnc(S)nc3)=O)o2)=O)CCC2(CNC(=O)N2)C1 C1(CNC(c2occ(C(=O)OC)c2)=O)CC(F)CN1C(C1(C)CC(C)(C)C1)=O N1(C(C2CN(C(=O)NC)C2)=O)CCN(C(=O)Cc2ccsn2)CC2(CC2)C1 C(CC(CC)C(=O)NCC1CC1CC(N1CCC(N(C)C)C(C)C1)=O)=CC C1(C(C)(C)C)CN(C(=O)Nc2cc(C(F)F)nn2-c2ccccc2)CCS1(=O)=O C1(NC(C=CC=CCC)=O)CN(C(C2CC2C#N)=O)C2CCCC12 N1(C(C(c2ccc(C)s2)C)=O)CC2CC(NC(=O)CCN(C)C(C)=O)C1C2 Cc1cc(C)c(NC(=O)C(C)NC(=O)Cc2occc2C)cc1C c1(CC)cc(C)c(C(=O)NCC2CCN2C(=O)CS(=O)(=O)NC2CC2)o1 c1(OC)cnc(Cl)[nH]c1=NC(CNC(C1CCC2CCCCN12)=O)C(C)C(C)C C=CCCCCCCCC(=O)N1CC(NC(=O)CCCCCN(C)C)C2CC12 C=CC1(CC)COCCN1C(c1cc(C(F)(F)F)ccc1Br)C(=O)NCC C1(c2n(C(CC)(C)C)nnn2)(NCc2cc(OC)n(C)n2)CCOC1C N1(C(C2CCN(C(=O)CCC3CC3)CC2O)=O)CCC12CCCOCC2 c1(CN(C(C2C(c3cc(C)on3)C2(C)C)=O)CC)ccc(OC)cc1 CC1CC2(CCC2)CN1C(=O)CC1CCCN(C(=O)CC23CCCC2C3)C1 C=Cc1cc(C(N2CC(CNC(=O)C(C)(C)C)CC23CCC3)=O)cc(F)c1 C1(NC(CCCC=C)=O)CN(C(c2c(C)coc2C)=O)CC12CC2 N1(C(C(C)OCCOC)=O)CC(C)(C)CC1CC(=O)NC1(C)CN(C(C)=O)CCO1 Cc1cc(C(=O)NC2CN(C(=O)C=Cc3ccsc3)CC2C)c(O)nc1C CC(C)(C)CC(O)C(=O)NCC(N1CCN(c2nnc(C(C)(C)OC)s2)CC1)(C)C C1(C)(C(N(CC(C)CNC(=O)C(c2ccc(Cl)cc2)CO)C)=O)CC2(CCC2)C1 C1(NC(C2(C)CC(=C)C2)=O)CN(C(c2csc(Br)c2Cl)=O)CC1C N1(C(c2c(OC)csc2)=O)CCN(c2ccccc2C(F)(F)F)CC1 C(=O)(C#CC(C)(C)O)N(C1CCCN(C(=O)COc2ccccc2)C1)C C1(N(C(=O)Cc2n[nH]c(=N)s2)C)CCCN(C(c2cc(C(F)(F)F)on2)=O)CC1 c1(C(=O)NCCC2(NC(CC3C(C)C3)=O)CCC2)cncn(C)c1=O C1(C(=O)NC2CCN(C(=O)CC3CCCC3)C2)CCCNS1(=O)=O C=CC(C)(CCOC)C(=O)N1CCCN(C(C2CN(c3nncs3)C2)=O)C(C)C1 N1(c2cccc(CC(=O)OC)c2)CCC12CCC(CN(C)C)CC2 C12(CNC(CSCC=C)=O)CCC(CN(C(c3cc(C4(C)CC4)n[nH]3)=O)C1)C2 c1(C(=O)NCCC2CSCCN2C(=O)CCC2CCCO2)ccc2ncnn2n1 c1(C(N2CCCCC2Cn2cc(CO)nn2)=O)cc2ccc(Br)c(Cl)c2s1 C(=O)(C1=NOC(C)(C)C1)N(CCSCC)C.C12CN(CCC1C)C(=O)CNC2=O.CC C(O)(CC(=O)NC(=S)NCCCF)(C(F)(F)F)c1ncc(C)o1 Cc1cc(Cl)cc(C)c1C(=O)NCC1CCN1C(C1(CCF)CC1)=O c1(C(=O)NC(CNC(c2c(C)nc(C)s2)=O)C(C)C(C)C)c[nH]c(C)c(Cl)c1=O N1(C(C(C)CN2CCOCC2)=O)CCC(NC(=O)CCN2CCC(O)CC2)C1C Cc1nnc2ccc(C(N3CCCN(C(=O)CC(F)(F)F)CC3)=O)cn12 C(=O)(CC(C)CCC)N1CCC(N(C(c2cncc(CC)c2)=O)CCOC)CC1 c1(C(=O)NCCOC2CCN(C(CC(C)c3cnn(C)c3)=O)C2)cn(C)[nH]c1=N C1(C(N2CCN(C(CNC(CC(C=C)(C)O)=O)=O)CC2)=O)Cc2nnc(C)n2C1 N1(C(CNS(CC)(=O)=O)=O)CCCN(C(=O)C=Cc2cscn2)CC1C(C)C c1(C(=O)NC2(CN(C(CS(CC)(=O)=O)=O)C)CC2)ccc2c(c1)CCCO2 O=C(C1=CC(O)C(NC(C2(O)CCOC2)=O)C1)NCCC(O)CCO N1(CC(=O)NCC2C3CN(C(c4cc(C)oc4C)=O)CC32)CCn2ccnc2C1 c1(CC(=O)NC(CNC(c2nc(C)[nH]n2)=O)CC(C)C)cnc(O)nc1O C(=O)(N1OC2CCC1CC2)C1C2N(C(c3c(CC)nc(C)o3)=O)CC(C=C2)C1 CCCC(C(O)C(=O)NC1CC2C=CC1C2)NC(C1(OC)CCCOC1)=O C1(NC(c2n[nH]c(C)c2C)=O)CN(C(c2ccc3c(c2)CCO3)=O)CC(C)(C)C1 C1(NC(CC(=O)NCC)=O)CN(C(c2csnn2)=O)C2CC12 CC1CC(C(=O)N(CCO)CC2CC2)CN(C(=O)CCc2ccnn2C)C1 C1(C2CC2)(C(=O)NC(CC)CNC(=O)CNS(=O)(=O)C2CC2)CCOCC1 c1(C(=O)O)ncc(-c2cn(CC(N3CCC(CO)C3)=O)nn2)cn1.C1CC1 c1(C(=O)NC(C=CC)C(=O)O)ccc(C)nc1N1CCCCC1 c1(CCNC(=O)CCNC(c2cnc(C3CC3)o2)=O)cccc(O)c1 c1(OC)ccc(I)c(C(=O)NCCN2CCN(C(=O)CCC(C)C)CC2)c1 c1(CCC(=O)NC2CC(NC(c3cc(C)ncc3)=O)C2)ccc2c(c1)CCCO2 C#Cc1ccccc1CC(N1CCCC(F)(C(=O)NCC(C)(C)SC)C1)=O C1(CN=c2nc(CCNC(C3CCCSS3)=O)[nH]s2)CC2(C1)CC1(CCC1)C2 Cn1nc(CNC(=O)CNC(=O)CCc2cnn[nH]2)oc1=O N1(C(C2CCSCC2)=O)CCCC(C2CN(C(C34CCN(C3)S(=O)(=O)C4)=O)C2)C1 CCC(C)C(C(=O)N(C)CCC1CCCCN1C(=O)Cc1ccc(O)nc1)OC N1(C(C2CCN(CC)CC2)=O)CCC(O)C(C(N2CCC2)=O)C1 c1(CC(=O)NC2(CO)CN(C(=O)OC(C)(C)C)C2)cnc(O)n(C(=O)O)c1=O CC1CCOCC1(F)NC(=O)CC1CCCCC1 CCCS(=O)(=O)CC(=O)NC(C1CCN(c2cc(O)nc(O)n2)C1)C N#Cc1cc(C(=O)NCC2CCN(C(c3ccc4c[nH]nc4c3)=O)C2)cc(F)c1 CCCC(CNC(C1(Br)CC1(C)C)=O)NC(=O)CCn1cc(C)cn1 C1(C(=O)NC(C(=O)NCC(=O)NCCOC)C(C)C)CCCCC1(C)C c1(NC)c(C(=O)NCC2CCCCN2C(=O)CCC2CC2)sc2nccnc12 N1(C(CCN(C(C2C=CC=CC=C2)=O)CC)=O)CCOC2CCC12 N1(C(C2(C#C)CCCC2)=O)CCC2(CCN(C(C3(C(F)F)CC(=C)C3)=O)CC2)C1 C=C(C)C(CC(=O)N1CC2CC2C1C(N1C(CO)CCC1CO)=O)OCC N1(C(C(C=C)(C)CC)=O)CCCCCC(NC(c2ccc(CN(C)C)nc2)=O)C1 N1(C(C2(C#N)C(C)C2)=O)CCCC2(CCCN2C(=O)C=CC2CCOCC2)C1 C(C(=O)NOCC(C)O)(c1ccoc1)NC(C1(COC)CC1)=O c1(C(=O)NCC(C)OC)ccc2c(c1)C1(CCCC1)CN2C(=O)C(C)CN c1(C(N2C3CC(CN(C(CNC(N)=O)=O)C3)C2)=O)cncc2cnccc12 C#Cc1cnn(CC(=O)NC2CCOC(C(=O)N(C)Cc3ncc[nH]3)C2)c1 N1(C(C(C=CC)O)=O)CCC2(CCCC2CNC(c2cc(C(N)=O)[nH]n2)=O)CC1 C(=O)(CC(CNC(=O)CC1CCCC12CC2)OC)NC(C#C)CC1CCCC1 N1(C(c2c(SC)cnn2C)=O)CCC2(CC2NC(c2cc(O)ncc2F)=O)C1 CCC(C(=O)NCC1CN(C(=O)CCc2cccc(O)n2)CCCO1)C(F)(F)F CN1C(=O)NCC12CN(C(C13CC(NC(=O)CC4CC5CCC4C5)(C1)C3)=O)C2 c1(C(=O)NC2CCCCN(C(C3CC4(CCOC4)C3)=O)C2)cccc2ncnn12 N1(C(CN(c2cccnc2)C)=O)CCN(C(=O)C(O)P(C)(C)=O)CC1C1CC1 N1(C(C(c2cccnc2)OC(C)C)=O)CC2CCC1CN2C(=O)CC1CC(=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1C(CN(C(C23OC(C)(C)C(C2)C3)=O)C2CC2)CCC1 c1(C(=O)NC2C(NC(C(C=C)CC)=O)CCC2)cc(O)ccc1Br N1(C(CC2ON=C(C)C2)=O)CCC(C)(C(=O)N(C)Cc2ccoc2C)CC1 C(CO)(CCCCNC(c1ccc(-c2ccccc2)nc1)=O)NC(CC(C)O)=O c1(OC)cc(OC)c(C(=O)NC2CCC(Nc3ncc(Br)c(OC)n3)C2)cc1Br C1(CNC(=O)CC(C(F)F)N2CCOCC2)CCc2ncccc2C1 C1(NC(C(C)OCC#C)=O)CCCCCC1C(=O)NC(c1c[nH]ccc1=O)C c1(C(N2CCN(C(CC3CC(=O)C3)=O)C3C2C3)=O)[nH]c2ccc(F)cc2c1Cl c1(C(N2CC(=C(CNC(c3ccc(C)nn3)=O)F)C2)=O)nnn2c1COCC2 CC(C)(C)CCC(=O)C(=O)N1CC2(COC(CNC(=O)C#CC3CC3)C2)C1 CC1(C)COCC1C(=O)NCCC1CCN(C(C2(c3cccnc3)CCC2)=O)C1 CC1CCCN(C(=O)C=C(Cl)Cl)C1.C12CCC(O1)CN(C)C2=O CCC(C)C(=O)C(=O)N1CCCC(F)(CNC(c2ccc(F)s2)=O)C1 CN1CCc2ccc(NC(C3CCCN(S(=O)(=O)C(F)F)C3)=O)cc2C1=O N1(C(c2c(C)c(N)n(C)n2)=O)CC2(CCN(C(c3ccncc3)=O)C2)C1 C1(CNC(CCC2OCC(C)(C)C2)=O)(NC(C2CC3CC2C3)=O)CCCCCC1 C(=O)(CCCCCN=[N+]=[N-])NCCC(C)(C)NC(c1ccccn1)=O CC1CCN(C(=O)ON2CCN(C3CCCC3)CC2)CC1COC(C(C)(C)C)=O c1(OC)cc(C2(C(=O)NCC3CCN3C(=O)C(F)C3CCC3)CCC2)ccc1C C1(C(N2CCCC2CO)=O)C2CC3C1C3C2CC1CCC1 CCC(CC(=O)N1CCCCC(CNC(=O)CC2OCCCO2)C1)C(C)C O=C(CCC(F)(F)C(F)F)NCC(C1CCC1)NC(=O)CC1(O)CCCCC1 C1(NC(C(CN(C)C)NC(C#CC(C)C)=O)=O)CCCCC12CC2 C1(COC)(CNC(=O)CNS(C)(=O)=O)CCCN1C(c1ccoc1Br)=O CC(C)(CO)C(CO)NC(C1CCOCCN1C(=O)CC1CC2CCC1O2)=O c1(C(N2C(C(N3CC(C)OC(C)C3)=O)CCCC2)=O)c(Br)cc(Br)c(Cl)c1Cl CC(C)(C)C(=O)CCCC(=O)N1CC(c2ccccc2)(NC(c2cc[nH]n2)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)N1C(C(C)NC(=O)CCCn2cccn2)CCCC1 N1(C(C(=O)NC(C(C(F)(F)F)OC)C)=O)CC2(CCC(=O)N2)C1 c1(C(=O)NCCC(C)NC(=O)CCC2CC2)nc[nH]c2nccc1-2 N1(C(C(C)=CC)=O)CCC2(CCC2NC(=O)CCc2cccnc2C)CC1 Cc1c(C(N2CC3CCC(C2)N3C(C2CCCC23CC3)=O)=O)cnc2ncnn12 CN1C(=O)CSC1=CC(=O)NCC(O)CCNC(c1ccc(-c2cccs2)s1)=O C1(C(N(C)Cc2cn(CC)nc2)=O)CCC=CC1NC(=O)CC1CCCOCC1 c1(C(C)(C)C)nc(-c2nc[nH]n2)sc1NC(=O)COC(=O)CN1CCCC1 C1(C(N2CC(C)(NC(C3CC(OC)C3)=O)C2)=O)CCCCC1C(N)=O N1(C(c2n(C)ccn2)=O)CCC(C)(CCNC(C2CC3CC3C2)=O)C1 C=CC(CC)CC(=O)N(CC(=O)NC1CCCNC1=O)C(C)C c1(N2C(C(=O)Nc3c(Cl)cc(F)cc3Cl)CC2)ncnc2cnccc12 c1(C(c2cn(CCNC(C3CN(C(C)=O)C3)=O)nn2)=O)cc(Cl)ccc1Cl Cc1ccc(S(=O)(=O)CC(C)NC(C2(c3nnnn3C)CC(C)N(C)C2)=O)cc1 N1(C(c2c(C)c(Cl)ccc2)=O)CCN(C(=O)CCCC#N)C(C#N)C1 c1(NC2CCCC(NC(c3occ(C)c3)=O)C2)cc(O)nc(O)n1 c1(CNC(C(C2CN(C(c3cc(C)[nH]n3)=O)C2)O)=O)c(C)nn(C)c1C c1(CCCC)nnc(C(C)NCc2ccn(CC)n2)o1 CCC(C(=O)NCC(C)(C)CNC(C1CC2(CCCC2)C1)=O)C(C)O S(=O)(=O)(c1cccc(Br)c1F)NC1CCCN(C(CC=C)=O)C1 c1(C(=O)NC(CC)CNC(C2CCS(=O)(=O)C(C)C2)=O)[nH]c(C)c([N+](=O)[O-])c1C Cc1cnc(N2CCC(CC(C)NC(c3cc(C(C)(C)C)[nH]c3C)=O)CC2)nc1 C(CC(=O)NOCCC(F)F)N(CC#C)C(c1ccc(C2CC2)o1)=O Cc1c(Cl)c[nH]c(=NCC2CN(C(C34CC(C3)C4)=O)CC23CCOCC3)c1C#N C1(C)(C(=O)Nc2c(SC(COC)C)cnc(Cl)c2)C2Cc3ccccc3C12 C1(CNC(Cn2c(C)ccn2)=O)CC2CCC(C1)N2C(=O)Cc1cc[nH]c1 C(CC(O)CC(=O)NCC(C)(C)CC1CN(C(=O)CC2(C(F)(F)F)CC2)C1)SC c1(C(N2CC3CN(Cc4ccc(OC)c(Br)c4)C3C2)=O)cccc(Br)c1C#N c1(C(N2CC(CC(N3CCC(COC)(NC(C)=O)C3)=O)C2)=O)cccc(C)c1F C1(NC(c2ccc(CCC)s2)=O)CCN(C(c2snnc2C)=O)CC1C(C)C c1(OC)cc(CC(C)N)cc(C(F)(F)F)c1.c1(C(CCCO)C2CCS2)ccccc1 Cc1ccc(C(=O)NCC(N2CCN(C(c3cnco3)=O)CC2)C(F)F)c(C)c1 C12CC3CCC(C1)N3C(=O)C1CN(C1)CC(=O)N2.C1(C)(CC)CCCC1C(=O)O c1(OC)cc(OC)c(C(=O)N(C)CCN(C)C(c2cc(O)ccc2C)=O)c(F)c1 c1(C(=O)NC(CNC(C(=O)NCC)=O)(C)C2CCC2)cnc(C(F)(F)F)c(Cl)c1 CC1CN(C(c2cnc[nH]2)=O)CC(CCNC(c2n[nH]cc2Cl)=O)O1 C1(NC(CC=C=C)=O)CCC12CN(C(=O)CC1CC(F)(F)C1)C2 C12CCC3(CN(C3)C1=O)O2.N#CC1CC(NC=O)C1.c1(N2CC(C=O)C2)cccnc1 CC1(C(=O)NC2C3CN(C(=O)Cn4cc(C5CC5)nn4)CC23)CC=CCO1 N1(C(C(CC(=O)O)NC)=O)CCC2(CC1)CC2C(=O)Nc1cnc(Cl)nc1 C(CCC(=O)NC1CCC1CNC(C1CCCO1)=O)SC C1(NC(C(C)OCC2CCCO2)=O)CCN(C(=O)CCCC2CCC2)CC1CO N1(C(C2C(C)(C)COCC2)=O)CCC(C2CCN(Cc3cocn3)C2)CC1 CC1(C(=O)NCCCNC(=O)Cn2cnc(=N)[nH]2)CCc2ccccc2C1 c1(C(N2CC(NC(CNC(=O)OC)=O)C(C)CC2)=O)noc(C(C)C)c1[N+](=O)[O-] C#Cc1ccc(F)c(C(=O)NCC(C(=O)OCCC)OC)c1.C(C)(C)(C)S C1(Cn2cc(CN(C)C(C3CN4CCN3CC4)=O)nn2)Cc2ccccc2O1 C1(C(C)NC(CC=CCC)=O)CCCN1C(c1conc1C1CC1)=O c1(COCC)nc(C)c(C(=O)N(CCCCNC(c2cnc(C)o2)=O)CC)s1 N1(C(C=C(C)C(C)C)=O)CCN(C)CC1C(=O)NC1CC1c1noc(C)n1 C1(CNC(N(CC(CC=C)O)C)=O)COCCC1(F)F C1(NC(C2CC(OC)CN2C(=O)C2=CCCC2)=O)CCN(C)CC1C N1(C(C=CC=CCC)=O)CCSCC1CCNC(C1COCCN1CCCC)=O N1(C(C=C(C)CNC(C2CCCCO2)=O)=O)CC2CC2C2CC12 C1(NC(=O)COCC2CCCC2)CCCC1NC(c1ccnn1CC(F)F)=O N1(C(c2ccccc2Cl)C)CC2CC(NC(c3ocnc3C3CC3)=O)CC1C2 N1(C(CCN(C(c2c(OC)n[nH]c2)=O)C(C)C)=O)CC2(C1)NC(=O)NC2=O CC(C)(C)C(C#N)C(=O)NCCC1(O)CCN(C(C2CCC3(CCC3)C2)=O)CC1 C(=O)(C(C)C(=O)N(CC(C)CNC(c1c(Cl)cnn1C)=O)C)OC c1(NC(C(=O)NCC23CC(COC)(OC2)C3)=O)cnc2c(c1)S(=O)(=O)NC=N2 c1(OC)cccc(CC(O)C(=O)N2CCC(NC(c3ccc(C)o3)=O)C2)c1 CCCCCCC(=O)NC1CC(CCC(=O)N(C2COCCC2O)CC)C1 C=CCCCC(c1nnnn1CC1CCOCC1)N(C(CC)C1CCCC1)C1CC1 CCS(=O)(=O)c1ccc(CC(=O)NC2CC3CCC(C2)N3C(=O)C(C)O)cc1 CC(CCOCc1ccccc1)C(=O)N(C)CC1CCC(NC(=O)OC(C)(C)C)C1 Cc1cc(F)c(NC(=O)C(O)CCCNC(=O)Cn2cnc(=N)[nH]2)cc1F c1(CCNC(C2CC(SC)C2)=O)cnc2ccccn12.C12(CCC(C)C1)C(=O)N2 C(=O)(CC(C)C(F)F)N1CCC(N(C(c2cnn(C)c2)=O)CC)CC1 C(=O)(CCCCCCCC1CC1)NC12C(CN(C(c3c(C(C)C)con3)=O)C1)C2 C(=O)(C1=NOC2(CCC2)C1)NCCSCC(N1CCC(C)SCC1)=O C(=O)(CCC(=O)N1CCCC(C(N2CCCC2C(N)=O)=O)C1)OC C1(NC(C(CC)(C)C)=O)CN(C(=O)Cc2n[nH]c(C)n2)C(C)(CC)C1 CC(C(=O)NCC1(NC(=O)C(C)(C)Oc2ccc(F)cc2F)CC1)C(C)C(C)(C)C Cn1cnc2c1CCCC2C(=O)NCC1CN(C(c2n[nH]cc2F)=O)C1 C12(CNC(c3c(C)ccnc3)=O)CCCC1CCN2C(=O)CCc1nccn1C n1(CC(=O)NC23CCC2CN(C(=O)CC24CCCC2C4)C3)nc(O)ccc1=O C1(C(N(CCOCCNC(C2CC(C)(CC)C2)=O)C)=O)OC(C)(C)OC1(C)C C12(CSc3ccc(C(=O)NCC4(C)N(C(C)=O)CCC4)o3)CC1COC2(C)C N1(C(c2c(C)ccc(F)c2)=O)CCc2oc(C(=O)O)cc2C1 CC(Cc1cnn(C)c1)C(=O)NC1CC(CCNC(C2(F)CC2C)=O)C1 n1(CC(=O)NCC(CC)NC(C2C=CC=CC=C2)=O)cc(Cl)c(O)nc1=O C(=O)(C(C)(C)S(C)(=O)=O)N1CC(C)C(NC(c2cncc(Cl)c2Cl)=O)C1 C12(NC(CCSCC(C)C)=O)CCN(C(c3cc(C(C)(F)F)n[nH]3)=O)CC1C2 c1(-c2cn(CC(=O)NC(c3n(C)cnc3)CC#N)nn2)cncc(C(=O)O)c1 C1(NC(c2cc(CC)on2)=O)CCC(C(=O)NCCC2CCCCO2)CC1 CC(C)C1=NOC(C)(C(=O)NC2CCCC2NC(c2cnc(O)c(F)c2)=O)C1 C1(C(=O)NC(C2OCCN(C(CSCCCC)=O)C2)C)CCC2(CC1)CC2(F)F c1(CC2(CS(=O)(=O)Oc3ccccc3)CC2)ccc(F)c(F)c1 N1(C(C2C(CC)C2)=O)CCCN(C(c2ccc(F)c(F)c2C)=O)C(C)C1 N1(C(C(C(C)OC)NC(C2CC(=C)C2)=O)=O)CCn2cc(C)nc2C1 C1(C(C)C)CN(C(C2CCCCC2CNC(C2(C#N)CC2)=O)=O)CCCO1 C1(C(=O)NCc2ccns2)(CNC(C(CC)N(C)C)=O)CCCCC1 c1(CC)nc(C)cc(=NCCCCC(C)NC(c2ccc(Cl)cc2C)=O)[nH]1 C1(OC)CCN(C(=O)C(C2(O)CCC2)NC(=O)C=Cc2cc[nH]c2)CC1(C)C C1(C(=O)NCC2N(C(C3(SCC)CC3)=O)CC(C)CC2)CC(C2CCCC2)C1 N12CC3COCC3(C1)NC(=O)C2C1CC1Cl.N1(C(CC(C)(C)C)C2CC2)CCOCC1 N1(C(c2c(CCC)n[nH]c2)=O)CC2C=CC1C(C(=O)NCc1cccnc1F)C2 C1(Nc2c(C(=O)OCCc3c(C)n[nH]c3C)cccc2)CCc2ncccc2C1 c1(C(=O)NCCCNC(CC2CC(CC)C2)=O)sc(Cl)c(Cl)c1N C(C(C)(C)C#CC(=O)NC1C(O)C2CCOC12)NC(c1ccc(OC)cc1)=O CCC(C)(C)C(C)CC(=O)NCC1CCCC1NC(c1cc(F)ccc1N)=O c1(C(N2CC(C#C)N(C(=O)C(C)N(C)C(C)=O)CC2)=O)ccc2cccnc2n1 c1(NC(C2CC(CCNC(CC(C)OC)=O)C2)=O)cc(C)c(O)cc1C C12CCC(CC1)NC(=O)N2C.C12CC(C1)NC(=O)N2.C(C)(C)(C)C1CC1 N1(C(C2CCN(C)C2)=O)CC(NC(c2cn(C)nc2C2CCCO2)=O)CC(F)C1 c1(C(=O)OCc2nnc(C)n2C)ccc2c(c1)nc(O)n2C c1(CCC(=O)NCC2CCN(C(C34CCC3C4)=O)CC2)cncc(F)c1 c1(C(=O)NCC2CCN(C(C3N(C)CC3)=O)CC2O)ccc2cnoc2c1 N1(C(C(CCCCC)O)=O)CC(NC(C2CC2c2cncs2)=O)CC12CCCC2 CCCC(C)(C)CC(=O)NCC1CN(C(C2CCCN2C)=O)CC1C C1(OC)CN(C(=O)CCn2ccnn2)CC1NC(=O)C(CCSC)N(C)C C1(n2cc(C(C)(C)OC)nn2)CCC(C(=O)NCc2cscn2)CC1 Cc1ncc(C(N2CCCC(n3ccc(C(F)(F)F)n3)C2)=O)cc1C(F)(F)F N1(C(C=Cc2c(C)n[nH]c2)=O)CCC(C2CC2)(NC(C2CC2(F)F)=O)C1 N1(C(C(=O)NC(C2CCCCC2)C(=O)C=O)=O)CCCC2(C1)CN(C)C(=O)O2.CN C1(CNC(=O)CNC(C2(SCC(=O)C3CC3)CC2)=O)CCCO1 N1(C(C(C(C)C)NC=O)=O)CC2CCC(C(=O)NC(c3cn(C)cn3)C)(C2)C1 Cc1cc(CC(=O)NCCNC(c2ccc(F)cc2)=O)cnn1 c1(C(=O)NCC2CCCC2NC(c2cnsn2)=O)ccc(Br)c(C(F)F)c1 N1(C(C(C=C=C)C)=O)CCC(C(=O)N(C)Cc2nccs2)CC1(C)C c1(C(=O)NCCC2CC(C(=O)N)C2)cc2c(C3CC3)cccc2[nH]1 c1(N(C)Cc2cccc(Br)c2)nc(N2C3CCC2CC3)c2c(n1)CCS2 C(c1cnc(O)nc1O)=CC(N1CCC(O)(C(C)NC(c2nc(C)[nH]n2)=O)C1)=O c1(CCC)[nH]nc(C(N2CC3(C2)CN(C(C2(CO)CC2)=O)C3)=O)c1[N+](=O)[O-] C(C)(C(=O)OC)NC(=O)NCCNCCC c1(CC(N2CCC(Cn3cc(COC)nn3)C2)=O)ccccc1Br c1(C(=O)NCC(C)N(C(Cc2cc(CC)no2)=O)C)cc(Cl)cc(Cl)c1OC N1(C(CS(CC)=O)=O)C(CNC(=O)CCOCC(F)F)CC2CCCC12 C1(c2ccccc2)COCCN(N2CC3(C=CCO3)C2)C1 n1(CC(CN(C2CCCCC2)CCCC)C)cc([N+](=O)[O-])cn1 C(=O)(CC(CC)CCC)N1C(CNC(CCC)=O)CC(F)C1 C12(OC)CCCC(C(=O)NC3CC4(C3)CC4NC(=O)CCS(C)(=O)=O)(CC1)C2 c1(CCC)csc(CNC(c2cc(Br)cs2)c2nnnn2CC2CCCO2)n1 C(=O)(CCN(C(=O)CCC1CCC1)C)N(CC#C)CCO C1(C(C)C)C(NC(c2cc(C3CCC3)[nH]n2)=O)CCN1C(C1(C(F)(F)F)CC1)=O c1(CC)cccc(OCC(N2CC(NC(c3ncsc3C)=O)C(C)C2)=O)c1 Cc1cccc2c1OCC2C(=O)N1CCN(C(=O)CC#N)CC12CCC2 c1(OCC(=O)NC2CCCN(C(c3c(C#C)c[nH]n3)=O)C2)cccc(CC)c1Cl c1(OC)ccc(CN2CCCC(NC(c3c(OC)noc3C)=O)C2)cc1 C1(C(N2C(CCNC(CCOCC#C)=O)CCC2)=O)CCOCC1(C)C c1(C(=O)NCCC2CC(NC(C3CCC3(F)F)=O)C2)cn(CC2CCCO2)nn1 c1(OC)ccc(CC(=O)NC2CC2C(=O)NCc2ccc(F)c(OC)c2)cc1F c1(C(=O)OC)ccc(C(C)C(N2CCN(C(=O)CSCC3CCCO3)CC2)=O)cc1 Cc1ccccc1C(C)CC(=O)NC(c1ccccc1)CNC(c1[nH]cnc1C)=O N1(C(c2cn(CC)nc2)=O)CC2(CNC(c3cnn(C)c3N)=O)CCC1CC2 c1(C(N(C)CC2CN(C(C3(COC)CCCCC3)=O)C2)=O)cnc2sccc2c1 n1(CC(=O)NC2C(C)CN(C(c3ccsc3)=O)C2)c(=O)nc(O)c2ccccc12 C1(C(N2CC(C)(NC(C3CCCS3)=O)C2)=O)CC2CCC1C2 C(C(C)CCCC(C)C)NC(CC1(C)CCN(C(C(CC)n2ccnc2)=O)C1)=O C#CCC(C(=O)N1CCCC(=C)C1)NC(c1nonc1CC)=O CC(C)C(O)C(=O)N(CC(O)CNC(c1cc(C#N)on1)=O)C C(=O)(C(C)(C)CCF)NCCCCC(=O)NC(CC(C)C)C Cn1nc(C(=O)NCC(F)CNC(C2(C)CCCS2)=O)c2cc(F)ccc12 N1(C(COC(C)C)=O)CCN(C2CCN(C(=O)C(c3ccc(O)cc3)=O)C2)CC1 C1(C(N2CCC(NC(C(CC)CN(C)C)=O)(CF)C2)=O)CCCCC(=O)N1 c1(CC)cc(C(=O)NC(C)(CNC(=O)CCCC2CCC2)CO)on1 c1(C(=O)NCC2N(C(C3C(C)OCCO3)=O)CCC2)nn(C)c2c(=O)[nH]cnc12 N1(C(c2c(CC)nccn2)=O)CC(NC(=O)CCc2cn(C)nn2)C(C2CC2)C1 CC1(C)CC(CNC(c2cncc(Cl)c2Cl)=O)N(C(=O)Cn2ccnn2)C1 c1(N2CC(=C(CNC(=O)CCC(=O)NCC)F)C2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CC(C)(CC(=O)N1CC2CC2(CNC(C2CCCCC2(C)C)=O)C1)C(F)(F)F C=CC(C)(CC)C(=O)N1CC(CN2N3CCN(CC3)CC2=O)C1.C(CCCCC)OC c1(SC)nc(N2CCC(NC(c3cnn(CCO)c3C)=O)C2C2CC2)cc(C)n1 C=CCC(C)(C)C(=O)NCCC1CCCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1 Cc1cc(C(=O)NCC(=O)NOCCN(C)C2CC2)c(C)[nH]1 N1(C(C2(C#N)CCC2)=O)CCC2CCC(C1)N2C(c1ccc2c(c1)CC(=O)N2)=O C1(C(=O)NCC(CN(C(=O)C=CC=C(Cl)Cl)C)O)CCc2nc(C(C)C)cn2C1 Cc1cc(C)c(-c2cn(CC(N3CCCC4OCCC34)=O)nn2)cc1C N1(C(c2c(OC)nn(C)c2)=O)C2CCC1CC(CNC(=O)C(F)C(C)(C)O)C2 N1(C(C(C)NC(C)=O)=O)CC(NC(c2ccc(CS(C)(=O)=O)o2)=O)C2CC2C1 c1(CC)cccc(C(N2CCCCC2c2nccs2)C(=O)NC2CCCC2)c1F C1(C(N2CC3(C(C(=O)OC)C3)C2)=O)CC(O)CCN1C(=O)CCc1cncnc1 c1(C(=O)NC2C3CN(C(C(CCCC)CC)=O)C2C3)cnc2c(=O)[nH]ccc2c1 c1(C(N2CCC(NC(c3cc4occc4s3)=O)(CF)C2)=O)cc(=O)cc(Cl)[nH]1 N1(C(CC(=C=C)C)=O)CC2C=CC1C(C(=O)NCCC(C(C)C)OC)C2 C1(O)(CNC(C(Cc2cc[nH]n2)NC(C(F)=CCC)=O)=O)CCN(C)C1 N1(Cc2ccc(C(=O)OCC)[nH]2)CCC2C(CCN2C(=O)Cc2cccnc2)C1 c1(C(=O)NCCN(CCOC)C(C23COCC(C2)C3)=O)cccnc1C1CC1 C1(C(N(CCCO)CC)=O)CC12CCN(C(c1cc(CC(C)C)nc(O)c1)=O)C2 C(=O)(C1=C(Cl)CCC1)NCC1(C(=O)NC2CCCC2N=[N+]=[N-])CC(=C)C1 c1(C(N2CC(NC(CN(C(C)=O)C)=O)C3C2C3)=O)cccc(Cl)c1Br C1(C(=O)OC)(CNC(N2CCCC(N(C)C)C2)=O)CC1S(C)(=O)=O c1(COC)ncc(C(N2CCC(C(C)NC(c3cc(C#N)c[nH]3)=O)C2)=O)c(O)n1 CC1CCC(Cl)=C(C(=O)NC2CCCCC2NC(c2ccc(N)c(F)c2F)=O)C1 C1(CC(=O)N(CC(C)O)C(C)C)CN(C(C2CCCC(O)C2)=O)CC1C c1(C(=O)OCC)ccc(C2C(=O)N2C2CC2)cc1.c1(CNC)ncc[nH]1 N1(C(c2ncn(CC)c2)=O)CCC(C2CCCN(C(=O)C(C)CC)C2)CC1 C1(CCC)(C(=O)OCC)CCCN1C(C1(NC(=O)CCC2CCCC2)CC1)=O N1(CC(=O)N(C2CCN(C(=O)C(O)CC3CCCCC3)C2)CCC)CC(C)(C)C1 C1(C(=O)NCCCOCC)C(C2CC2)CCN1C(C1CCCCC1)=O N1(CCC)CC(C(=O)N(CCCCCNC(=O)C(C)n2cccn2)C)CC1=O C(C)(CNC(=O)C=C(Cl)Cl)(CNC(c1cccn1C)=O)OC C(CN=c1[nH]cc(C#N)c2ccsc12)N(C(C(c1ccc(F)cc1F)C)=O)C C1(NC(CC2(N(C)C)COC2)=O)CCOCC1NC(C1COCCO1)=O Cc1cnc(C(=O)NCC2CC(NC(c3n[nH]c(C)c3Cl)=O)C2(C)C)cc1Cl C1(CC)CCCN(C(=O)Cc2cn(C)cn2)C1C(=O)NC1CC2OCCCC12 c1(NC(C2N(C(c3c(C)nns3)=O)CC(F)C2)=O)cnc(C)c(C#N)c1 CC1CCCc2c(C(N3CC4CCC4(CNC(=O)C=C4CCC4)C3)=O)cnn21 C1(CNC(COCCOCC)=O)CC12CCN(C(c1cscc1OC)=O)CC2 c1(SC)nc(CNC(c2ccc(SC)o2)=O)cs1 C1(CC(N2CC(NC(c3c(CC)nco3)=O)C(C)C2)=O)CCOCC1(C)C c1(NC(C2N(Cc3n(CC)ccn3)CC(O)C2)=O)cccc(C)c1C c1(C(=O)NCC2N(C(C3C(C)C3)=O)CCCC2)cccc(Br)c1O N1(C(C(c2ccc(F)cc2)C)=O)CCN(C(C2CCC(=O)O2)=O)C(CC(F)F)C1 Cc1cc(O)ncc1C(=O)NC1CN(C(=O)C(N2CCC(C)C2)=O)CCC1F C1(C(C)NC(C2(C(N)=O)CC2)=O)CCCN1C(c1ccc(Cl)[nH]1)=O O=C(CCC(=O)Nc1ccc(Br)cc1)Nc1nccs1.C12CC1COC2=O C1(C(=O)NCC2CCCN2C(C2(C)CCC(C)C2)=O)(NC(C)=O)CCC(C)CC1 C1(C(N2CCC(CN(C(=O)C=Cc3cc[nH]n3)C)CC2)=O)CCc2nn[nH]c2C1 C12=C(C(F)(F)F)NC(=NC3C4CC3CN(C4)C1=O)C=C2.c1(C(C)=O)c[nH]cc1Br C1(CNC(c2cnsc2)=O)CN(C(c2cnc(O)c(Cl)c2)=O)CC2(CCC2)O1 C1(C)(C(=O)NC(CC(=O)NCC(NOC)=O)CC2CC2)CC2CCC1C2 CCC(C)(CC)C(=O)NCC1CC2(CC(NC(C3(CC)CCCO3)=O)C2)C1 C12(NC(C3N(CC)CCCC3)=O)CCC(NC(c3cscc3OC)=O)(CC1)C2 c1(NC(C(C)NC(CNC(CNC(C)=O)=O)=O)C)ncnc2cc(Br)sc12 N1(C(c2c(SC)nn(C)c2)=O)CCOCC1(C)c1cn(-c2cnn(C)c2)nn1 C1(NC(CC(C)C2CCCO2)=O)CC2(CCN(C(C34CC5CC3C4C5)=O)C2)C1 c1(NC2C(NC(c3c(OC(C)C)ccc(Cl)c3)=O)C2)ncnc2ccc(F)cc12 C1(NC(C(CCO)OC)=O)CN(C(c2cccc(F)c2C)=O)CC1(C)C CN1C(=O)C2CC1CCN2C(c1cnc(Cl)s1)C(=O)NCC1CCCO1 C1(C)(C(=O)OC)CN(C(=O)OC(C)(C)C)CC1(F)F.C12(C)CC(C1)C2=O.C(=O)C(F)(F)F C1(CC=C)(NC(=O)C=Cc2cn[nH]c2)CCCN(C(=O)C(c2ccccc2)O)C1 C1(C)(CC)C=C(C(=O)N2CCC(CN(C(c3cc(=O)n(C)o3)=O)C3CC3)CC2)C1 CC1C(C(=O)N2CC(CC(=O)N(CC3CC3)CC3CC3)C3(CC3)C2)=NOC1C c1(C(C)C)nccc(=NCC2(C(N3CC45CCC4(COC5)C3)C)CC2)[nH]1 C(=O)(C1CCCc2nn[nH]c21)N1C(CNC(CCCC#C)=O)CC(OC)C1 C1(NC(C2(CC=C)CCN(C(c3c[nH]c(=N)o3)=O)C2)=O)CCCCCCC1 CC1CC(C(N2CC(C(c3ccccc3)C3CC3)C2)=O)C12CCC2 c1(C(N2CC(C)(NC(CC3C(CC)C3)=O)C2)=O)cc2c(OC)ccc(C)c2[nH]1 c1(C(N2C(C)(C)C(NC(C3CC(CF)C3)=O)CC2)=O)cc(Cl)cc(Cl)c1O N1(C(C(C)N(C)C)=O)C2CCC1CC(NC(=O)Cc1nc(C(F)(F)F)nn1C)C2 c1(C(=O)NC2C(CC)CN(C(=O)C(C)=C3CC3)CC2)cn2cccc(Cl)c2n1 CC1CC(NC(C2(C)CCC(F)(F)C2)=O)CCN1C(=O)CCN1CCCC1 CC(=O)CCCC(=O)NC(CN(C)C)C(N1CCC(O)(CN(C)C)C1)=O c1(OCC)ccc(-c2ccc(CNC(=O)NC3CCN(C)C3=O)cc2)cc1C CC(CC1CC1)C(=O)NC(CNC(C1CC1c1ccccc1)=O)Cc1ccccc1 C(=O)(C(CO)C(C)(C)C)NCC(CNC(c1c(C)cco1)=O)CO C(=O)(C(C)C(=O)N1CCN(C2CN(C(c3sccc3OC)=O)C2)CC1)NCC C1(C)(COC)CC(NC(=O)CCCNC=O)CN1C(=O)CCCCCSC c1(C(=O)NCC2CCCN2C(c2ccsc2)=O)ccc2oc3ccccc3c2c1 c1(C(N2CC3CCN(C(C(C)c4cc[nH]n4)=O)CC32)=O)n[nH]c2c1CN(C)CC2 N1(C(CCOCCCNC(CC2CC(N(C)C)C2)=O)=O)CCCOC(CCO)C1 N1(c2nnc(C)s2)CCC(NC(c2ccnc(CN(C)C)c2)=O)C(CO)CC1 N1(C(c2c(CC)csc2)=O)CC=CCC1C(=O)NCC(Cl)=CCl c1(C(=O)NC2CCN(C(C(C=CC)O)=O)CC2O)c(C)c(C)c(C)c(C)c1C C1(Cn2cc(CCCC)nn2)CN(C(c2ccccc2OC(C)C)=O)CC12CC2 C1(NC(C(C=C)O)=O)C(C)(C)C(NC(c2ccc(F)c(C#N)c2)=O)C1(C)C Cc1cc(C)c(C(=O)N(CCCCN(C)C(C2(C#N)CC3CC3C2)=O)C)c(S)n1 N1(C(CN(C(C)=O)C)=O)CCN(CCNC(c2cc(C(C)(F)F)ccn2)=O)CC1 C(=O)(CCC1CCc2ccccc21)N1C(CN(C)C(c2cn(C)cn2)=O)CCC1 S(=O)(=O)(c1ccc(C(F)(F)F)c(Br)c1)NC(c1ccccc1)N(C)Cc1cnn(C)c1 n1(CCCC)cc(CNC(=NCc2cnc(SC)o2)NCC(C)C2CC2)c(C)n1 CC(C)CC(C)C(=O)NCC1CCCCCCC1 c1(CCC(=O)NC(CC(C)NC(c2c(CC)[nH]cc2)=O)C)ccc(Br)nc1 c1(C(=O)NC)cccc(C(N2CCOC(Cn3cc(-c4cncs4)nn3)C2)=O)c1 Cc1c(C(=O)NC2CC(CNC(C3(C)CCC(=O)C3)=O)C2)sc2ccc(F)cc12 c1(CNC2CCN(C(C3(O)CC3)=O)C2)c(F)cc(Cl)cc1Br CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1(CF)CCN(C(c2ccncc2C)=O)C1 c1(C(=O)NCCCN(C2CCCC2)C(C2CC(C)(C)O2)=O)ccc(Cl)cc1Cl N1(CCN(S(Cc2cccc(C)c2)(=O)=O)CC2CCCO2)C2CCC1CN(C)CC2 C#CC1(NC(=O)C=CC(C)NC(=O)CCCn2cncn2)CC(F)(F)C1 c1(C(N(CCOCCNC(C(CC#C)O)=O)C)=O)cc([N+](=O)[O-])nn1C C1(C2CCN(C(=O)CSCCC(C)C)CC2)(NC(Cc2nc(C)[nH]n2)=O)CCC1 N1(C(C(CC2CC2)OC)=O)CC(C)C(C)(CNC(=O)C(C)(C)NS(C)(=O)=O)C1 c1(NC(COC)C(C)C)nc(N(C)Cc2ccc(SC)cc2)nc2scnc12 C(=O)(C1=CCCOCC1)N1CC(C(=O)Nc2cnc(SC)nc2)C2(C1)CC2 C1(C2(O)CN(C(=O)CC(n3nc(C)cc3C)C)C2)(CNC(CCC(=C)Cl)=O)CC1 n1(CCCC)ncc(C(=O)NCCC2CC(NC(C34CCCC3C4)=O)C2)c1C CC1C(NC(=O)C2=CCOC2)CCN1C(C1CCN(C(=O)N(C)C)CC1)=O C1(NC(Cc2c(C)n[nH]c2)=O)CCN(C(c2cnc(C(F)F)s2)=O)CC12CCC2 c1(NC(C(=O)NCC(c2ccccn2)(C)C)=O)cc(F)c(F)cc1N c1(COCCN(C(C#CCCC)C)c2ccccc2)ccc(F)c(OC)c1 N1(C(C(=O)N(C)C)=O)CC2(CCN(C(c3cc4n(n3)CC3(CC3)C4)=O)CC2)C1 N1(C(C(C2CCN(C(c3c(CC)nccn3)=O)C2)F)=O)CCCN(C)CC1 CCC(C(=O)N1CCC(C(C)NC(=O)CC2COCCN2C)C1)C(C)C C1(COC)(OC)CCN(Cc2nnn(C(=O)OC)n2)CC1 C#CCC(CC(=O)NCC(=O)NCCO)NC(c1c[nH]c(=NC)o1)=O C1(C(N(CC)CC2CCCN2C(c2coc(Cl)n2)=O)=O)CCC(F)(F)C1 Cc1cc(C(=O)NC2C=CC(CNC(C3(C(N)=O)CCC3)=O)C2)ns1 Cc1cc(C)c(C(=O)NC2CC(C)N(C(c3sccc3C#N)=O)C2)cn1 c1(CCCC(=O)NCC(C)(C)NC(c2n(C)cc(Cl)c2)=O)ccc2c(c1)OCO2 c1(NC(CCCc2cccc(C(C)=O)c2)=O)ccc(F)c(Cl)c1.C1(=O)C(C)O1 Cc1cc(=NC(=O)C(=O)N2CCC(C(C)NC(C3(Cl)CC3)=O)CC2)[nH]o1 c1(CC(=O)N(C2CC(NC(C(F)=CCC)=O)C2)C)csc2sc(C)cc12 C(=O)(C1=CCCC(C)(C)C1)NCC(CC)(CC)NC(C(CCC)CC)=O c1(C(=O)NC2C(CNC(=O)CCOC3CCC3)CC2)ccn(-c2ccccc2)n1 c1(SCC)cccc(C(=O)NC2CCN(C(C3CCC(=O)C3)=O)C2CC)c1 N1(C(c2cnc(C(=O)OCC)s2)=O)CC2(C1)C(C(=O)OC)CCS2(=O)=O C12CCC(=O)N1C2=O.c1(N(C)C)ncc(C(=O)NCCOCCSC)s1 C1(C(N(CC(F)C2CCC2)C)=O)CN(C(c2ccc(C#N)o2)=O)CC12CC2 c1(C(=O)NC2(CNC(CC(CC)NC(C)=O)=O)CC2)cc2ccc(CO)cc2[nH]1 C1(NC(C(Cc2c(C)cccc2)C)=O)C(C)(C)C(NC(c2ccon2)=O)C1(C)C n1(CC(=O)NCC(C)NC(c2cccc(S(C)=O)c2)=O)ncc2cccnc12 c1(CC)ccsc1C(N1CC(CNC(=O)Cc2ncc(C)[nH]2)(CC2CC2)C1)=O c1(CN(C(CC2CCCCO2)C(=O)O)C=O)cc(F)c(Br)cc1F N1(CC)CCCCC1C(=O)NCC(C1CC1)N(C(=O)CCC1CCCC1)C C=CCC(CC(F)F)NC(C1CC(C)CCN1C(=O)C=Cc1cocn1)=O N1(CC)CCC(NC(C2C3CCC(C3)N2C(C2(OC)CCC2)=O)=O)C(C)C1 C1(NC(c2c(OC)nn(C)c2)=O)CC1C1CCCN(C(=O)C=Cc2ccoc2)C1 c1(C(N(C2CN(C(C3(C)COCCO3)=O)CC2O)C)=O)ccn2c1CSCC2 c1(C(N2C(CN(C(CC(C)N(C)C)=O)C)CCC2)=O)cc(C2CCC2)nn1C C1(CN(C(CC=C=C)=O)C)CCCCN1C(C1CCCN(C(=O)OCC)C1)=O C1(C(N(C2C(C)COCC2)C)=O)CCCCN(C(=O)CC2CC=CC2)C1 c1(C(=O)NCC2OCCCN(C(c3c(C)ncnc3)=O)C2)cccc2cc[nH]c12 N1(C(c2cc(C)[nH]c2)=O)CC2CCCN(C(C3CC4CC(O)C(C3)C4)=O)C2C1 c1(SCC)ccc(C(=O)NC23CC(NC(c4scnc4C)=O)(C2)C3)cn1 C1(C(=O)NC2C(C)COC2)CC(O)CN1C(=O)CCC(=O)N(C)C N1(C(C2C(OCC)C2)=O)CCCCC1n1cc(CCCS(N)(=O)=O)nn1.C(CO)O c1(OC)c(C(=O)NCC(C)N(C(=O)C(C(C)C)NC(C)=O)C)ncnc1C n1(CCC)ccc(C(=O)NCCC(C)NC(=O)C(C)(O)C2CCC2)n1 OC1CCCC(NC(c2ccc(C(F)(F)F)cc2)c2ccccc2)CC1 C(=O)(C1=CCC(C)CC1)NCCC(C(C)C)NC(=O)CC(c1cccc(F)c1)C C12(CNC(c3cc(CC)ncc3)=O)CCC(CC1)N2C(c1cnc(Cl)[nH]1)=O C1(C(=O)NC2CC3CC3C2)CCN(C(=O)CCOCCCOCC2CC2)CC1 N1(C(CCSCC)=O)CC(CNC(C2CC3(CCOC3)C2)=O)C2(CCOCC2)C1 C#Cc1cnn(C)c1C(=O)NC1CCN(C(c2ccnc(C)c2N)=O)CC1C C(C)(CCC(=O)NCc1cc[nH]c1C(=O)NCC1CC1[N+](=O)[O-])OCC N1(C(C23CC(C)(C2)C3)=O)CCOC(CNC(c2cccc(CCC#N)n2)=O)C1 c1(NC(C=C2CCN(C(c3cc(C)nn3C)=O)CC2)=O)cc(Br)cc(Cl)n1 N1(C(C(c2n(C)ncc2)O)=O)CCC2(CCCN2C(=O)C=C2CCC2)C1 C1(C(=O)NCC2CN(C(CN(CCOC)C)=O)C2)CC2CCC1CC2 C1(C(=O)NC(C#N)C(N)=O)CCCC12CCN(C(c1cccc(Cl)c1Br)=O)C2 c1(CC)ccsc1C(=O)N(C1CC(NC(c2cnc(CC(C)C)s2)=O)C1)C C(=O)(CC(C)C(C)C)N1CC(CNC(CCSCC(C)C)=O)OCC1 c1(C(=O)OCC)nc(Cl)ccc1NC1(C)CN(Cc2ccccc2)CC1C c1(C(=O)NC23C(CN(C(CCCC)=O)C2)CCC3)cc([N+](=O)[O-])cc(C)n1 C1(CNC(C=C(CCN(C)C)Cl)=O)CCCN(C(=O)COC2CCOCC2)CC1 c1(C(=O)NCC(C)CNC(=O)CC2CSCCO2)c[nH]c(=O)cn1 c1(C(=O)NCC2C(C(=O)NCC(C)(C)OC(C)C)C2)cc2ccccn2c1 C1(C)(NC(C(CCC2CC2)NC(c2c(CC)n(C)nn2)=O)=O)CCC(C)(C)C1 N1(C(c2ccc(C#C)o2)=O)CCCC2CN(C(C3(F)CCOC3)=O)CCC12 c1(C(N(C)CCNC(C2(F)CC=CC2)=O)=O)ccc2ccc(Br)cc2n1 CCC(C(=O)NCC1NC(=O)CNN1)NC(N)=O.C1(C(=O)NC2CC2)CCCO1.SC Cc1cc(C(N2CCC(C)C2CNC(=O)CCc2cn(C)nc2C)=O)[nH]c1C N1(C(c2ccc(C)s2)=O)CC(CNC(C2C3CCN2CC3)=O)C(O)C1 C1(C(=O)NCC(CCNC(=O)CN2CCC(C)(C)C2)OC)CCOCC12CCC2 c1(C(=O)NC2C(OC)CN(C(c3cn(CC=C)nc3)=O)C2)ncnc2ccsc12 c1(CC(=O)NCc2c(C)cc(OC)nc2)ccc(F)cc1[N+](=O)[O-] N1(C(C2(OC(C)C)CCOC2)=O)CC2CC2(CNC(=O)C=CCO)C1 N1(C(C(c2ccccc2)OC)=O)CC(NC(C2(F)CCOCC2)=O)C(C)C1 C1(NC(C=CC(c2ccccc2)C)=O)CCN(C(C2SCCCS2)=O)C(C)C1 C=Cc1cncc(C(N2CCOCC2C(N2CCN(C)CC2CC)=O)=O)c1 N1(C(C2(C#C)CC2)=O)CC(CC(=O)N(C2CCCCC2)CC)C(C)C1 c1(SC)cc(C(=O)NCC2(NC(C3CC3c3cccs3)=O)CC2)c(C)o1 CCC(C)C(O)C(=O)N1CCCCC1CCNC(c1n[nH]cc1F)=O C(=O)(C(CC)C(=O)NCCCCNC(C1COCCN1C)=O)OCC C1(CC(C)NC(c2cn(C3CC3)cn2)=O)CCN(C(C2C3(CC3)C23CC3)=O)CC1 Cc1cc(=O)c(NC(C2C(O)CCN2C(=O)C2=CC3C=CC2C3)=O)c(C)[nH]1 N1(C(C#CC(=O)N(C)C)=O)CC2CCCC2(NC(=O)Cn2nc(O)ccc2=O)C1 CCC(C)(CNC(C1(CC)CCN(C(c2ncccn2)=O)C1)=O)CC c1(C(=O)NCC(CNC(c2c(CC)n(C)nc2)=O)OC)cnc(Cl)cc1N C=CCC(C)(C)CCNC(C1CC(NC(=O)C(C)COC(C)=O)C1(C)C)=O c1(C(=O)NCC2N(C(C(C)(O)C3CCC3)=O)CC2)ccc(Br)nc1 c1(C(N2CC(NC(=O)CCF)C3C2C3)=O)ccc(N(C2CC(F)(F)C2)CCO)nc1 N1(C(c2nn(C)cc2Br)C(=O)NCC(c2ccccc2)OC)CC2CC=CC1C2 C1(NC(c2ccc(C(F)F)cc2)C)CCCN(Cc2ccccc2)C1=O C1(CN(C)C)CCN(CC(C2COCCO2)=O)C1 O=C1CC(C(=O)NC2CN(C(c3cn4ccnc4s3)=O)CC2O)NC(=O)N1 c1(OC)cccnc1C(C)NS(=O)(=O)CC1(CC(F)(F)F)CCOCC1 Cc1cccn2c(CC(=O)NC3CC(CCNC(=O)C(C)(F)F)C3)cnc12 C1(N(CC(N2CCC2CNC(=O)Cn2ncn(C)c2=O)=O)C)CCC(=O)N(C)C1 CC1CCCN(C(=O)C=Cc2cscn2)C1CCNC(C1CC=CC1)=O C1(O)(C(C)(C)C)CCN(C(=O)NCCOCCOc2cccc(Cl)c2)CC1 C1(N(C(CSCC#C)=O)C)CCC(NC(c2ccsc2C(F)F)=O)CC1 N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2cc(C(C)C)n(C)n2)=O)C2CC12 C#Cc1ccc(C(=O)NCCC(C)NC(=O)CC23COC(C)(C2)C3)c(F)c1 Cn1ccc(CC(=O)NCC2CC2CNC(=O)CC2CSCCS2)c1 c1(CC)ccc(Cl)c(C(=O)NC2CCC2NC(=O)C(C)(C2CC2)OC)c1 Cc1cc(C)c(C)c(C(=O)NC2CCCC(N(C(=O)Cn3nccn3)C)C2)c1C c1(NC(C(C)(C)NC)=O)ccc(NC(=S)NCC(C)C)cn1 C1(CCNC(C2CCC=CO2)=O)CCCCN1C(c1ccc(-c2cccs2)s1)=O c1(-c2c(OCC(=C)C)cc(F)cc2)ccc2[nH]cc(C#N)c2c1 C1(OCC)CCCC(C(N2CCC2CNC(=O)COc2ccccn2)=O)C1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(C(C)C)CC(=O)NC(C)(CO)C(C)C C1(NC(=O)NCCCc2n(C)ncc2)CCCC=C1Br C1(CNC(CSCCCC)=O)CCN(C(=O)COCc2ccccc2Cl)CC1C C1(NC(CCSC)=O)CC2(C1)CC(C(=O)N(CC(O)CF)CC)C2 C=C1CN2C(=O)CCC2(C(=O)NC(C)CCN(C)C(C2CC(=O)CC(=O)N2)=O)C1 N1(C(=O)NCCC2CCN(C)C2)CCOC(c2nccs2)C1 c1(C(=O)NC2C(NC(=O)Cn3cnc4ccccc34)C2)cc2cc[nH]c(=O)c2s1 N1(c2nnc(-c3ccc(C)c(F)c3)n2Cc2cnn(C)c2)CCn2cncc2C1 C=CCC(CC(F)F)C(=O)N1CCC(NC(=O)Cc2cc[nH]n2)CC1C C1(CNC(C(CSC)O)=O)CN(C(C2(O)COC2)=O)CCC1(F)F c1(CC)c[nH]c2ncnc(N3CCC(CF)(CNC(=O)CC(=O)OC)C3)c12 C1(C(N2CC(O)(CNC(c3c(C)scc3)=O)C2)=O)CCN(C)C1C C1(CNC(C(C)c2ncco2)=O)CCC(NC(=O)CCC2CCOCC2)C1 CC1(C)C2CCC(C(N3CC4CC3C4NC(c3cccc4ccsc34)=O)=O)C1C2 C(C(C)C(C)C(=O)NCC(C1CCN(c2nccc(C)n2)CC1)(C)C)OC c1(CC(=O)NCCC2(CNC(c3cc(F)n[nH]3)=O)CC2)ccn(CC(F)(F)F)n1 c1(CC(N2C(C(C)NC(CCC(C)SC)=O)CCC2)=O)cc2ccccc2s1 c1(N(c2c(OC)cccc2OC)C2CC3CC2CN3)cc(Cl)nc(C#N)n1 c1(N2C(CN(C)C(C3CC4CC3C3CC43)=O)CSCC2)ncn(C)c(=O)c1Br CCCC(C)(C)C(=O)NC1CN(C(=O)CCNC(=O)Nc2ccccc2)CC1O C1(NC(c2n(C)c(O)nc2)=O)CC2CN(C(C3CC34CC4)=O)CC2C1 N1(C(c2nccc(C)c2)=O)CCC2(CCCC2NC(c2ccc(F)c(Br)c2)=O)C1 CCC(C)C(O)C(=O)NC1COCCN(C(c2c(C(F)(F)F)ncn2O)=O)C1 C1(CC#C)(C(=O)N(CC=C)CCF)CCN(C(c2coc(SC)c2)=O)C1 CC1COCC(CNC(=O)NCc2cccc(-n3cc(CO)nn3)c2)O1.CCO Cc1nn(C)c(C)c1CC(=O)NCC1C(C)CCCN1C(=O)CSCC(F)F N1(C(c2ccc(-n3ccnc3)nc2)C(=O)NCC)CCOC(C)C1(C)C c1(OCC(=O)OC)ccc2cccnc2c1CN1CCCC1C(=O)O.NCN N1(C(C(CC)CC)=O)CCCC2(C1)CN(C(C1CCC1C(=O)OCC)=O)C2 c1(CNC(C2C(C=C)C2)=O)ccc(CNC(=O)C(O)CC(C)C)c(F)c1 c1(C(N2C(CNC(C3CC=C(C)CC3)=O)CCCC2)=O)ccc2nnn(O)c2c1 c1(C(=O)NCC(c2cccc(OC)c2)NC(=O)C(C)CSC)c(N)ccc(C)c1F c1(C(C)O)ncc(C(=O)NC2CCC(NC(=O)COC3COC3)C2)s1 C1(C(=O)Nc2c(C(=O)OCC)cno2)CC2CC2N1C(=O)Cc1cccnc1Br N1(C(c2nnsc2-c2ccccc2)=O)CCN(C(C2(F)CCCC2)=O)C2CC12 C(=O)(C1CCCc2cncn21)NC1C(SC)CN(C(=O)C2=CCCCC2)C1 N1(C(CCCOCCOCC)=O)CC2CC1C2NC(C1CCC(F)CC1)=O c1(C(=O)OC)cc(NS(=O)(=O)CC2CCS(=O)(=O)C2)c(O)cc1F C(CCCC(=O)N(C1CCN(C(c2ncn(C(C)C)n2)=O)CC1)C)OC c1(OC)ccc(F)c(S(=O)(=O)NC(c2cccc(F)c2)C(=O)OC)c1F C(CCC(=O)OC(C)(C)C)N(CC(F)F)C.C1(c2ccsc2)C(=O)N1CCO C1(O)(CCNC(=O)C(O)C2CCC2)CCN(C(=O)C(F)=CCCF)C1 C(=O)(C(F)(F)C(C)(C)C)N1CCC(N(C(CC2C(C)=NN(C)C2=O)=O)CCO)C1 c1(-c2n(C)ccn2)ccc(C(=O)NC2C3CC(NC(=O)CC4CCC4)CC23)cc1 N1(C(CCc2c(C)nccn2)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)C2(CC2)C1 CN1CC(C)(C)CC1C(=O)NC1CC2(C1)CN(C(C1CNC(=O)N1)=O)C2 Cc1nn(C)c(I)c1C(=O)NC1CCC1NC(c1cnco1)=O C1(C(=O)NC(C2CCN(C(c3cnns3)=O)C2)C)(CC#N)CCCC1 n1(CC)cnc2c(NCCCN(C)C)[nH]c(=NC3CCOC3C)nc12 C1(NC(CCC=CC(C)C)=O)CN(C(=O)CC2CCC(F)(F)C2)CCC1CO c1(OCCC)ccc(C=CC(=O)NCCC(C(=O)O)OC)cc1OCC.OC C12(CC)CN(C(C3(C)CCOC3C)=O)C(CNC(=O)C=CC(C)(C)SC)(C1)C2 C1(N(C(C2(NC(=O)OC(C)(C)C)CC2)=O)C)CC2(C(=O)NCC(N)=O)CC12 Cc1nnc(C(C)NC(=O)CNC(c2cn[nH]c2)=O)s1 C1(C)(C(N2CCC(N(C)C(c3ccncc3Br)=O)C2)=O)CC(C2CC2)=NO1 N1(C(C(C)Sc2ccccc2)=O)CCCC(O)(CNCC2CN3CCC2CC3)C1 N1(C(C(CC)N(CC)CC)=O)CC2CCC1C(NC(C1CCCSC1)=O)C2 C(=O)(C(CC(C)C)N(C)C)N1C(CN(C(CCCOCC=C)=O)CC)CCCC1 c1(C(=O)NCC(CCNC(c2n(CC)ncc2)=O)O)c(Cl)c(C)nn1C N1(C(C(C)N(C(CSCCC)=O)C2CC2)=O)CCC(C)(O)C1 c1(CC(=O)NCC(CC=C)NC(=O)CCCCC(C)C)cn2c(n1)CCCC2 C1(NC(N2CC(CC)OC(CC)C2)=O)Cc2c[nH]cc2S1(=O)=O CC1C(C)N(C(C2CNC(=O)O2)=O)CCN1C(=O)CCC(F)(F)F C#CCC(C)C(=O)NC1CC(OCCSC)C1(C)C C1(C(=O)OCC#C)CCCC1=C1CC1NC(C1CC1NC(=O)NCC)=O.OCC c1(N(CCCN(C(C(c2ccc(Cl)cc2)C)=O)C)C)nccnc1F N1(C(CC#N)=O)C2CCC1CC(NC(c1cc(S(N)(=O)=O)c[nH]1)=O)C2 Cc1cc(=NC(=O)C2(F)CN(C(C3CCC(=O)N3C)=O)C2)[nH][nH]1 C1(CCC)CN(C(=O)CSC(F)F)CCN1C(=O)Cc1ncsc1Cl CSC1=C(C(=O)N2CC3(C2)CN(C(c2cccc(C)c2)=O)C3)CCCC1 C(C(CO)C(F)(F)F)C(N1CCC(C)(c2ccc(C(F)(F)F)cc2)C1)=O C1(C)(NC(C(C)(C2CCC2)NC(CC=C)=O)=O)CC(O)(CO)C1 N1(C(C2C(CC)OCC2)=O)CCCC(NC(=O)C=C2CCCCC2)C1C CC1CC(C(=O)N(CCC(=O)O)Cc2ccc(F)cc2)CCS(=O)(=O)C1 C1(CNC(c2ccc(COC)s2)=O)COCCN1C(c1cc(CF)on1)=O c1(C(=O)NC(C(CO)NC(c2c(SC)scc2)=O)C)ccc2cc(C)ccc2c1 c1(C(N2CCCC(NC(c3c(C)[nH]nc3Cl)=O)CC2)=O)cn2cccnc2n1 Cc1nn(C(C)(C)C)c(C)c1C(=O)NCC(CC(C)C)NC(=O)CC1CC1(C)C Cc1ccc(C(=O)NC(C(=O)NCC(C)Cc2cccs2)c2ccco2)s1 CC(CC(=O)N(CCC(C)(C)NC(c1cnc(C2CC2)s1)=O)C)CC(C)(C)C C#CC1(C(N2CCS(=O)CC2C)=O)CCN(C(c2nnsc2N)=O)C1 C1(CC(N2CC(CCNC(c3cccc(Cl)c3)=O)(OC)C2)=O)CCC(C)(O)CC1 c1(OC)ccc(C(=O)NC(C2CN(C(c3nc(C)n(C)n3)=O)C2)C)cc1F C1(C(=O)NCCc2ncn(CC)c2)N(C(=O)C(C)SC)CC12CCCC2 Cc1cc(C)c(C(N2CCCC2C2(NC(c3sccc3Cl)=O)CC2)=O)o1 C#Cc1cn(C)nc1C(=O)NC1CCN(C(=O)CCN(CC)CC)C(C)C1 CCCCCCCCCC(C)CC(=O)N1C2CCC1(CNC(C1CC1C)=O)CC2 CN1CCN(c2ccc(C(=O)NC3(CNC(C4CC=CCC4)=O)CC3)cn2)CC1 c1(N(CCCN(C)C(c2ccc3nccn3c2)=O)C)nc2cccc(F)c2s1 Cc1nc(NC(C2CCN(C(c3ncc(Br)cc3Cl)=O)C2)=O)ccc1Br N1(C(C2(C)CCCN(C(c3ccc(F)cc3F)=O)C2)=O)CC2CC(O)CC1C2 c1(CN(C(CN(C(=O)C(C2CCOC2)OC)CCC)=O)C)ccn(C)n1 N1(C(C=CCC)=O)CC2CCC(C1CO)N2C(=O)Cc1n[nH]cc1Br C1(C(N(CCCN(C(=O)CC2CCC2)C)C)=O)CCCC12CC2 c1(C(=O)NCC2C=CC(NC(CCOCC)=O)C2)ccc2c(c1)NC(=O)NC2 c1(C(=O)NCCCc2cccc(F)c2Br)nc(Br)n2c1CCCCC2 c1(C(=O)NC2C3(C)CC2N(C(c2cccnc2S)=O)C3)cnc2ncccn12 Cn1c(O)nc2cccc(NC(=O)NCCC3CCC4(CCC4)O3)c12 C1(CC(=O)NCCOCCCN(C(=O)Cc2ccns2)C)COCCO1 C=Cc1ccc(C(=O)NC2CC(CCC(=O)NCC(C)(O)CO)C2)cc1 c1(CC)cc(C(=O)NC2CC(N(C)C(c3cc(CF)on3)=O)C2)ns1 c1(CCC(=O)OC(C(=O)OC)Cc2cccnc2)ccncc1C C12(C(=O)NC3(CC=C)CN(C(=O)CC(CC)OC)C3)CC3CC1(CO)CC3C2 C(=O)(C(C)CC(=O)NC1CC(NC(=O)CCn2cc(Cl)cn2)C1)OC c1(C(=O)NC2(C)CC(NC(COCCC)=O)C2)nccn2nccc12 C12(NC(=O)Cc3cscn3)CCCC1CN(C(=O)C(c1cscn1)NC=O)C2 C1(NC(c2cnc(Cl)s2)=O)CN(C(C2CC3(CCCC3)C2)=O)C2(CCC2)C1 C1(NC(c2ccc(SC)s2)=O)CC12CCC(NC(=O)C(C)NC(N)=O)CC2 C1(C(=O)NCC2(C(N3CC(OCC(C)C)C3)=O)CCC2)CCCC(C)(C)C1 c1(C(=O)NCC(C2CCCN2C(c2cnns2)=O)(C)C)ccc(N)cc1Br N1(C(C2N(C(c3cccnn3)=O)CCN(C)C2)=O)CCC2(CNC(=O)C2)C1 c1(C(=O)NC2CC(C(=O)Nc3c(C)nsc3)C2)c(C)ccn1C N1(C(C2ON=C(C)C2)=O)CC(C)N(C(C2CCCC2)=O)CC1C c1(C(N(C2CCCC2)CCNC(C2CCCN(C)C2)=O)=O)cc2ccsc2n1C C(C(C)(O)C(=O)NC1CC(C(C)NC(C2(C)CC2(F)F)=O)C1)OC C(CC(CC)C(=O)N(CC(C)CNC(c1cccc(C)n1)=O)C)=CC C=CC(C)(CC)C(=O)N1CCCCC(CNC(=O)Cn2nc(O)ccc2=O)C1 Cc1cc(Cl)nc(Cl)c1C(N1CC2CN(C(c3cccc4ccoc34)=O)CC12)=O C(=O)(C(C)C(C)C(C)(C)C)NC1CN(C(Cc2nc(C)sc2)=O)C2(C1)CCC2 C(=O)(C1=Cc2cccc(OC)c2OC1)N1C2CCC(NC(CC=C)=O)(C2)C1 c1(CC)ccccc1NC(=O)NCC1(C(=O)Nc2cccc(OC)c2)COC1 CC1OC2(CO)CC1(C(=O)NCC1CCCN(C(C34CCC(CC3)OC4)=O)C1)C2 c1(CSCCOC(c2ccc(C3CCCO3)cc2)=O)cc(=O)n2ccsc2n1 c1(C(=O)NC(c2cccc(N3CCCC3=O)c2)C)cc(O)nc2c(Br)cccc12 N1(C(CC(=O)NCC)=O)CCC(NC(c2onc(Br)c2C)=O)CC1 C1(CC#C)CN(C(C23CC(NC(C4CCN(C)C4)=O)(C2)C3)=O)CCO1 C(c1ccc(SC)cc1)=CC(N1CC(COC)(CNC(C2CCN(C)C2)=O)C1)=O c1(C(=O)NC(Cn2cc(-c3cccc(OC)c3F)nn2)C)ccc([N+](=O)[O-])cc1 n1(CC)cc(NC(c2cccc(F)n2)=O)c(C(=O)Nc2ccc(SC)s2)n1 c1(C(=O)NCCc2ccc(OC)cc2)cc(Cl)ncc1NCc1cnc(C)nc1 Cc1cc(C(=O)NCC2CC(C(=O)NCCc3cncs3)=NO2)cc(F)c1 CCC(C)(C(=O)NCC1(CNC(=O)CCSc2ccccc2)CCC1)C(N)=O C1(O)(CC(=O)NC2(C(=O)NCC3CCC3)CC(CO)C2)CCOC1 N1(C(CCCC(=C)C)=O)CCCCC(C2CN(C(C3CCOC3C(C)C)=O)C2)C1 C1(C(=O)NC(C2(C(=O)NC3CCC(F)(F)C3)CC2)C)COCC1(C)C C(=O)(C(O)CCS(C)=O)NCC12OCCC(NC(c3ccc(OC)s3)=O)(C1)C2 C=CCC(C(=O)OCC)NC(=O)C(Cc1ccoc1)NC(c1coc(NC)n1)=O C1(CNC(C2CCC(COC)C2)=O)CC(C)(C)CN1C(c1cc(F)ccc1N)=O C1(NC(NC(CC)CCC=O)=NCC(C)F)CCc2cc(OC)ccc2C1.OC Cc1nccn1CCC(=O)NCc1n[nH]cc1C(=O)NCC(F)Cl N1(C(CC=CCC)=O)CCN(C(=O)C(C)=C)CC(C)(C)C1 C1(NC(C2(F)CN(C(CC3CN(C(C)=O)C3)=O)C2)=O)CCCN(CCO)C1 c1(C(=O)NCC(c2cccnc2)NC(CSCC=C)=O)ccc2c(c1)CC2 N1(C(C2(C)CCCCCC2)=O)CCC2CCC(C1)N2C(=O)Cn1cnccc1=O C1(F)(CNC(c2c(OC)ccs2)=O)CCN(C(c2cnc(SC)s2)=O)C1 c1(C(=O)NCC2C(CNC(c3c(C(C)C)onc3)=O)C2)noc2c1COCC2 C(C(O)C(=O)NCC=CCNC(=O)Cc1csc(Br)n1)=CCCC CCC(CC)CC(=O)NC1CCC(N(C)C(C2CSCCS2)=O)CC1 N#CC1CCCN(C(=O)CC2CN(C(c3ccc(CN(C)C)[nH]3)=O)C2)C1 Cc1ccc(F)c(C(=O)N=c2ccn(C)[nH]2)c1[N+](=O)[O-] C12CN=C(NCCC1)N2.N1(C(C2CCOC2)(C)C)CCCC1=O c1(C(C(N2CC(C)C(C)C2C)=O)NC(c2cnc(C)nc2)=O)c(C)cccc1Br Cn1cnc2cccc(C(=O)NC3CCN(C4CCNCC4)C3=O)c12 c1(OC)cc(OC)[nH]c(=NC2CN(C(=O)CCc3ccon3)CC23CCC3)n1 N1(C(CCc2n(C)ncc2)=O)CCN(C(=O)CSc2nc[nH]n2)C(C2CCC2)C1 c1(C(=O)NC2CCCCN(C(CCC(=O)OC)=O)CC2)cnc2c(n1)CCCC2 CN1CC2CCCN(C(C3CCOCC3NC(=O)C=Cc3cncn3C)=O)C2C1 C(=O)(CC(C)(C)C)NCC1C(C(C)NC(C(C)NC(N)=O)=O)C1 Cc1ccc(C(CC(=O)OCC(=O)OC(C)(C)C)NC(=O)OC(C)C)cc1 c1(C(=O)NC(CCNC(CSCCC(C)C)=O)C)cc(N)ccc1F C(CCC(C)CC(=O)N1CC2CC1C2NC(c1cc2n(c1)CCC2)=O)=C(C)C C(=O)(C1=Cc2ccccc2C1O)NCCCNC(C(CC(C)C)C(C)C)=O N1(C(C(Cc2cnc[nH]2)C(=O)N)=O)CCCCC1c1cn[nH]c1.n1(CC)cnc(Br)n1 Cn1cc(C2CC2C(N2CCC(CCNC(c3ccnn3C)=O)C2)=O)cn1 C1(C(=O)NC(CC(=O)NCCNC(=O)NCC)(C)C)CCC(C2CC2)C1 N1(C(CN(C)C(N)=O)=O)CCN2CCN(C(=O)CCCc3cnn[nH]3)CC2C1 c1(C(=O)NC(C2CCCC2)CNc2cccc(C(N)=O)c2)cnn2ccsc12 C(CN=c1[nH]c2c(C)cccc2o1)N(C(C1CC(OC)C1)=O)C c1(-c2onc(COC)n2)sccc1C#N C(=O)(C1CCCc2nc[nH]c21)C(C1CC(N(C(c2n(C=C)ncc2)=O)CC)C1)=O N1(C(C=CCC)=O)CCC(NC(C2(C)CCCC2)=O)C1 Cc1ccc(C(=O)NCC2CC3CC(C2)N(C(=O)CC(F)(F)F)C3)c2c1CCC2 N1(C(C(C2CCCC2)OC)=O)CC(O)(CCNC(=O)C(C2CCOCC2)C)C1 C#CC1CCCC(CNC(C2(C#C)CCN(C(=O)CCC(F)(F)F)C2)=O)C1 C1(CNC(C2C(C)C2C)=O)CN(C(C2(c3cccc(Br)c3)CC2)=O)CC1(C)C c1(CCC)cc(C(=O)NCC(C)(CO)NC(=O)CCCc2ccccc2)n(C)n1 Cc1c(C(F)(F)F)n[nH]c1C(N1CCCC1CNC(C1(C2CC2)CCCO1)=O)=O C(=O)(CCCCCCC(C)C)N1C(CC)C(NC(=O)CN2CCC(C)CC2)CC1 N1(C(CC(n2c(CC)ncc2)C)=O)CC2(CC2)CC1CNC(=O)C(F)C(F)(F)F C(C1CCc2nccn21)NC1CC2(C(O)C2)C1 c1(CC(N2CCC(SC)C2)=O)cnc2n1CCOC2.C1(=O)C(C)(C)CN1C1CC1 c1(C(=O)NCC2(C)N(C(Cc3cc(C)on3)=O)CCC2)ccc(Cl)c2occc12 CCS(=O)CC(=O)N1C(C(=O)NCc2n[nH]cc2C)CC2CC12 c1(CC)c[nH]nc1C(N1CC(C(C)NC(=O)Cc2sccc2C)C1)=O C1(CNC(c2sccc2Cl)=O)CC2CCC(C1)N2C(C1CC(=C2CCC2)C1)=O N1(C(CN2CCC3CN(Cc4cc(C)[nH]n4)CC32)=O)CCc2ncc(Cl)cc2C1 c1(N2CCC(C(CC)C)CC2)cc(NCCC2CCCCC2O)nc(C)n1 c1(C(N(CCNC(C23CC(COC)(OC2)C3)=O)CCOC)=O)cc(F)ccc1Cl CCCC(O)CC(=O)NC(C)CCNC(=O)CCCOc1ccc(Cl)cc1 CC1(C)CC(=O)NC1CNC(N1CCC12CCC2)=O N1(C(C2COCC(C)(C)O2)=O)CC2CCCC(C1)N2C(C1SCCCS1)=O CC1CC(C(=O)NCCn2ccc(=O)cc2)CN(C(C2CC3CC2CC3O)=O)C1 CC(C(=O)OCc1ccccc1)C(=O)N1CCCC1CNC(=O)Cc1cn[nH]c1 Cc1sc(NC(C2(c3cccc(O)c3)CC2)=O)nc1NCc1cscn1 C(C)(C)(CC(=O)NCCF)N(C(C1OCC(C)C1)=O)C C(C)(CNC(=O)C(N)Cc1cc(Br)sc1Br)(C(F)(F)F)OC C1(C(N2CC(NC(CCCC#C)=O)C(SC)C2)=O)CCCC2(CCOCC2)O1 CC1(C)CCc2c(C(N3CCC3Cn3cc(CN4CCOCC4)nn3)=O)n[nH]c2C1 C1(N(C(c2nccn2C)=O)CC)CCN(C(=O)CCc2ccncc2Cl)CC1 c1(CC)cc(OC)cc(C(=O)NCC2CCC(NC(=O)C(C#N)C(C)C)C2)c1 Cc1nccc(C(N2CCC(C(C)NC(=O)CC3CC3)CC2)N2CCCC2)n1 c1(C(N2CC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)ccc2nccnc2c1 Cc1cccc2[nH]c(=NCC3CCCCN3C(=O)CCC(F)F)sc12 c1(C(=O)NCC2CCCC(NC(c3ccon3)=O)C2)ccc2sccc2c1 Cn1nc2n(c1=O)CCN(c1nc3nncn3cn1)C2 CC1(C(=O)N(CC(N2CC=CC2)=O)C2CC2)CCCN1C(=O)Cn1cnnc1O Cc1cnc(C(=O)NC2CC2NC(c2cccnc2C(=O)OC(C)(C)C)=O)nc1 C1(C(C(F)(F)F)(F)F)CC=C(CNCC(Br)Br)CC1 C12(C(=O)O)CC3CC(C1)CC(NC(C1C4CC4C4CC14)=O)(C3)C2 N1(C(c2c(C)csc2)=O)CCOC2CN(C(c3ccc(N)c(Cl)n3)=O)CC12 N1(C(C(C)N2CCC2)=O)CCC2(CC1)CC(NC(=O)CCCCC(N)=O)C2 N1(C(CNC(C=CC(C)C)=O)C(F)F)CCN(C(=O)C(C)O)CC1 N1(C(CC(COC)NC(=O)CC2(C)CCOC2)=O)CC2(CO)CCCC2(F)C1 CCCCC(C(=O)N1CC(O)(C(F)C(=O)Nc2ccc(OC)cc2C)C1)C(C)C N1(C(CC(C)SC)=O)CCN(C)C(C(=O)Nc2cnc(C)c(Cl)c2)C1 CC(C)CCC(F)C(=O)NCC1CCC(C(=O)NC(CO)C(C)(C)CO)C1 N1(C(CC(C)C)=O)CCCC2(CNC(c3cnc[nH]3)=O)CC12 C(=O)(CCCCCS(N)(=O)=O)N1CC(CNC(Cc2c(C)noc2)=O)N(C)CC1 c1(OC(C)C)cccc(C(=O)NC(C)(C)C(C)NC(=O)C=C(C)C(C)(C)C)c1 C1(OC)CCC(C)(C(=O)NC2CC3CCC2N3C(c2cc(C)cc(O)c2)=O)CC1 C1(C(=O)NCc2ncn(CC)n2)(CC)CCN(C(=O)C(CO)N(C)C)C1 C(=O)(C(C)(CC(COCCC=C)=O)NS(=O)(=O)CC)N(CCNNC(C)=O)C.C CC(C)C(C)(O)C(=O)NC1CC1NC(c1csc(C2CC2)n1)=O C(=O)(C(C)(F)C(=O)N(C1CN(C(=O)CCC2CCCN2C)C1)C)OCC c1(C(N2CCOC(Cn3cncn3)C2)C(=O)NCCCC)ccnc(Br)c1OC C(=O)(CC(O)C(C)(C)C)N(CCN(C(c1c(CC)nc(-n2cccc2)s1)=O)C)C CC1CC2(CCN(C(=O)C=CCN3CCCC3)CC2)CN1C(C1CCN(C)C1)=O N1(C(C(CCC)NC(C2CCCOCC2)=O)=O)CCC12CC(O)C2 C(=O)(CCP(C)(C)=O)N1C(C(=O)OC)CC(n2cc(Cn3ccnc3)nn2)C1 Cc1c(Cl)ccnc1C(=O)NC1CCC(C)(CNC(c2[nH]cnc2C#N)=O)C1 n1(CC)ncc2cc(-c3nc(-c4nccs4)nn3C)c(C)nc12 N1(C(C(CC)=CCCC)=O)CCC(C)(CC(=O)NCC(N2CCCC2)=O)C1 N1(C(c2ccc(Cl)cn2)C(=O)NC(CC)C)CCSC(C)C1C C(CCC(=O)NOCCOCC1CC1)(C(C)C)NC(Cc1nc(C)oc1)=O c1(C(N2C(C(=O)NC3CCOCC3O)CSCC2)=O)ccc2cc[nH]c2c1 CC1(C)CC(CC(=O)NC(C(N2CCCC23CC3)=O)C2CC2)CCO1 N#CC1CN(C(=O)C=CC2CC2)CC1N=c1nc2[nH][nH]cc-2c(O)n1 C(=O)(C(C)CC(F)(F)F)NC1C(NC(c2nc(C)n(-c3nc[nH]n3)n2)=O)C1 N1(C(C2CCC(C)C2)=O)CC(C2(NC(=O)CCN3CCCC3=O)CC2)C1 c1(CN)ncccc1C(=O)N(C1CCCCC1)CCO C12(NC(C3(OC)CCC3)=O)CC(CNC(=O)COC3CCCCCC3)(C1)OC2C Cc1ccc(C(C)CC(=O)NCCOCCN(C(=O)CSC(F)F)C)cc1 c1(C(N(CCCN(C(C(C(CC)O)(C)C)=O)C)C)=O)cc2c(cc1F)OCO2 C1(c2cn(C)nn2)CCCCN1N1CC2CC2C1.c1(C=O)ccc(-n2ccnn2)o1 C(=O)(CC1=NNC(=O)C1)N1C(CNC(C(C)SCC)=O)CC(F)(F)C1 C1(CNC(C2CCS(=O)(=O)CC2)=O)CN(C(=O)Cc2cscn2)CCC12CCC2 c1(C(N2CCC(N(C(c3cncc(CC)c3)=O)C)C2)=O)ccc(CO)cc1OC O=C(CCC(CF)CF)NC12CC(C(=O)NCC3CCOC3=O)(C1)C2 C1(NC(CSCC)=O)CN(C(=O)Cn2c(O)nnc2O)C(C)(C)C1 C1(C(N2CCC(NC(c3csc(C)c3C)=O)C2)=O)CCCN2CCCC12 N1(C(c2nccc(OC)c2)=O)CCCCC(CCC(=O)NC(C)C(C)(C)O)C1 Cc1nc2ccc(C(=O)NC3CCC(F)(CNC(C4SCCS4)=O)C3)cn2n1 c1(OC)ccccc1C(C)CC(=O)NC1CC1CNC(=O)Cc1ccsc1 c12ccc(cc1)CC(=O)N1CC(C1)O2.c1(SCC(=O)OC(C)(C)C)ccccc1 c1(C(N(CCNC(c2c(SC)scc2)=O)C)=O)cc(Cl)c(Cl)cc1C c1(C(N2CCCC3(CNC(CCCCC)=O)C2C3)=O)cc2ccnc(Cl)c2s1 C(=O)(CC(C)C(C)(C)C)NC1C(C=C)CN(C(=O)COc2ccccc2)C1 CCCCC(C)(F)C(=O)N1CC(F)CC1CN(C(=O)CC(C1CC1)C1CC1)C C(=O)(C1=CC2(CCOCC2)C1)N1CCC2CCN(C(C(CCC(C)C)O)=O)CC21 N1(C(CCC#C)=O)CCCC(O)(CNC(=O)COc2ccccc2C(C)(C)C)C1 C1(C(N2CC(NC(c3cn(CCO)nn3)=O)CC(C)C2)=O)CCCC12CCC2 c1(C(N(C)CC2OCCN(C(CCCC=C)=O)C2)=O)cc(C)ccc1[N+](=O)[O-] N1(C(C2C(c3cn(C)nc3)OCC2)=O)CCN(C(=O)OC(C)(C)C)C2CCCCC12 N1(CCC)CCCC(CNC(=O)C(=O)NC2CCCCC2OC)C1 O=C1OCCC1CCC(N1CCCC1Cc1cccnc1)=O C(=O)(C(C(=O)N1CCC(NC(C2CC(N(C)C)C2)=O)C1)C(C)(C)C)OCC c1(OC)cccc(Cl)c1C(=O)Nc1cccc(C(=O)NCc2c(Br)cnn2C)c1 N1(C(CC)=O)CSCC1C(=O)NCC=CCNC(C1COC1)=O C(=O)(CCCCN1CCCCC1)NCCC(NOC(C)C)=O.C1(=O)C(C(C)C)N1 N1(c2c(C(=O)OC)c(C)ccn2)CCN(C(c2occc2C)=O)CC(C)(F)C1 C(=O)(C1=COCCC1)NCCn1ncc(C(N(C)CC2OCCC2(C)C)=O)c1 c1(C(N(C(C)C(=O)N(C(C)CC(N)=O)C)CC)=O)nc(O)sc1C N1(C(c2[nH]c(=NCC)sc2)=O)CC(C2CCCN(C(C3(C)C=CCCC3)=O)C2)C1 CN1CCC2(CCCN(C(=O)C3=CCCC3)CC2)CC1 CCCCC(O)CC(=O)NC1(C)CCN(C(c2cc(C#N)n(C)n2)=O)CC1 C1(NC(CCOC(C)=O)=O)C2CCC1N(C(C1Cc3ccccc3S1)=O)C2 C(c1ccc[nH]1)=CC(=O)NCC1(C(=O)NCC2(CCOCC)CC2)CC1 N1(C(CCSC)=O)CCN(C(c2cc(F)ccc2F)=O)C(C)CC1C C1(CNC(C2CC(SC)C2)=O)CCN(C(=O)C(C2CCCCC2)O)CC1O C1(CNC(Cc2cc(C)no2)=O)CCCC2CN(C(=O)C=CCCC(C)C)CC12 C=C(C)CC(C)C(=O)NCC1N(C(c2cccc(CN(C)C)c2)=O)CCC1(C)C Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCCc2nccs2)c(O)c(C)n1 c1(C(C)C)ncc(C(=O)NCCC2CC(NC(=O)CCNC(=O)CO)C2)[nH]1 c1(C(CNC2CN(C(C(C)OCCOC)=O)C2)O)cccc(OC(F)F)c1 C(=O)(C#CC1(C)CCCO1)N(CCNC(c1cc(C(F)(F)F)cc(Cl)n1)=O)CC Cc1cccc(CC(=O)N(C)CCN(C)Cc2cn(C(C)CO)nn2)c1 N(C(=NCCN(c1ccccc1Cl)C)NCCC1(C)CCC1)C1C(C)C1 N1(C(C2CC=CCC2)=O)CC2CN(C(=O)C(c3ccccc3F)(F)F)CC(C1)O2 c1(C(C(=O)NC2CC2)N(C2CCCCC2)C)cncc(Cl)c1 c1(C(N2CC(C)(NC(CCC=C)=O)C2)=O)ccc(F)c(C)c1Cl N#Cc1cn[nH]c1C(N1CCCC(N(C(=O)C=CSc2ccccc2)CCO)C1)=O C1(C(=O)OCC)C(C(=O)NC(C)(C)C)C2COCC12.C1(C(=O)NC)CC(OC2CC2)C1 CC1OC(=O)NC1C(=O)N(CC(O)CNC(c1nnn(C(C)(C)C)n1)=O)C Cc1cc(C(=O)NCC2(CNC(=O)C(C)(C)CO)CCCC2)cc(C)c1 c1(C(N(C(C)C)CC)=O)cc(CO)ccc1NC(=O)CCc1cnn[nH]1 C(=O)(C(CC)C(=O)OC)N1CC(C=C)(CC(=O)NCC(C)C(=O)OC)C1 c1(SCC)ccc(NC2CC2)cc1.C12CN(CCO1)C(c1cscc1C)C(=O)N2 Cc1cc(C(=O)NC2CC3(C2)CN(C(C2CC2(C)C(C)C)=O)C3)ccc1O N1(C(CS(CC)(=O)=O)=O)CCc2ncc(NC(=O)C(C)Cn3cccn3)cc2C1 CCCC(CC)CCC(=O)N1CC2CC1C2NC(=O)COCC(C)C N1(CC(=O)NC2(CC=C)CN(C(c3cc(C(=O)OC)no3)=O)C2)CCP(C)(=O)CC1 C(c1ccccc1)=CCC(=O)NC1CCN(C(c2cccc(CO)c2)=O)C1 c1(C(=O)NCC(CNC(=O)CCC(F)(F)F)OC)cc(C#N)cc(C)n1 c1(C(=O)NC(C2CCOC2)CNC(C(C)=C2CCC2)=O)c[nH]c2c(F)cccc12 C1(CCC)CN(C(=O)C#CC(C)(C)C)CCN1C(=O)C(C)P(C)(C)=O c1(CC)cccc(CC)c1CC(=O)NC1CCN(C(=O)CC2CC3(CC3)C2)C1C CC(C)(CO)C(=O)NCc1ccc(C(=O)NC2CCC2(C)C)cc1 N1(C(C2(c3ccc(OC)cc3)CC2)=O)CC2CCC(C1)N2C(c1cncs1)=O Cc1ccc(F)cc1NC(=O)C(C)(C)NC(=O)CCc1ccccn1 N1(C(CC2CCCN(C(C)=O)C2)=O)CCCC(CCNC(=O)CSC(=N)N)CC1 C1(CNC(c2ccnc(Cl)c2F)=O)CC2(CCN(C(=O)CSC3CC3)CC2)CO1 C12(CNC(c3cnc(C)s3)=O)CCCCC1N(C(=O)CCC1(O)CCC1)CC2 C(=O)(C1SCCc2sccc21)NCCCOCCN(C(C(CC)(C)CC)=O)C N1(C(c2c(OCC)cccc2)=O)CCCC(C2CC2NC(=O)CSC(F)F)C1.OCC N1(C(C2C(=C)C2)=O)CC2CCC1CN2C(=O)CCCOc1ccc(C)c(C)c1 c1(C(N2CC(NC(C(CC)C)=O)CC(C)(C)C2)=O)c[nH]c2nccc-2c1C C1(N(C(CCC(=O)N(CCC)CCC)=O)C)CCN(C(=O)CC2CC2)CC1C N12CC3CC=CC(=C3C1)C(=O)C2=O.c1(NC(=O)NC(C)C)ccc(N(C)C)cc1 N1(C(C2CCC(C)(C)C2)=O)CC(NC(C2(n3cncn3)CC2)=O)CC(F)C1 C(=O)(C#CC1(CC)CC1)N1CCC(CNC(C(C)(C2(C)CC2)OC)=O)C1 c1(CN(C(CNC(c2c(C)nc(Cl)cc2)c2nccs2)=O)C)c(F)cc(Br)cc1Br c1(C(=O)Nc2c(C(N)=O)nccc2)cc([N+](=O)[O-])cnc1O C(C(C)(C)C(=O)NCCCCCCN(C)C(c1nc(C)sc1C)=O)NC(C)=O c1(OC)ccc(C)cc1-n1cc(CCC2CCCN2C(C2COC(C)C2)=O)nn1.O S(=O)(=O)(c1[nH]c(=NCc2ccc(C#N)o2)ccc1Br)NCc1c(C(C)C)con1 c1(C(=O)NC2CC(NC(CCCC=C)=O)C2)cc(N2CCNC2=O)ccc1Cl C1(CCOC)CN(C(C2CCC(F)(F)C2)=O)CCN1C(c1ncc(F)cn1)=O C(=O)(CC(C)(C)C#N)N(C)CC1CCN(C(=O)C(=O)NCC2CC2)CC1 CC1CC(C(=O)N(C(CNC(C2CCCC2C)=O)C2CC2)C)C(C)O1 Cc1nc(C(C)C)ccc1C(N1CC(C(C)NC(=O)CCc2cccnc2)C1)=O c1(C(C)C)cc(C(N2CC(O)(CNC(=O)CC3CC4CC4C3)C2)=O)ns1 CC(C)CC(C(=O)N1CC(S(C)=O)C1)ONC(C1(C)CCCOC1)=O CN1CCC(N(C(c2ccoc2CN(C(=O)CC2CN(C)C2)C)=O)CCO)C1 N1(C(CCOCC)=O)CC2CC1CC2NC(=O)C(C)Oc1cccc(Cl)c1 CC1CN(C(=O)Cc2cnccc2Cl)CCN1C(=O)C(COC(C)(C)C)N(C)C c1(OC)ccc(C)c(C(=O)NCCN(C(=O)C(C(C)(C)C)OC)C)c1N Cc1cnc(C(=O)NC(C)C(C)NC(=O)Cc2ccnc(O)c2)c(C)c1 Cc1ccc(C(=O)NC(CNC(=O)Cc2cccnc2C)C(C)C(C)C)nc1C c1(OCC)cnncc1NC(C12CC(C(=O)Nc3ccccc3C)(C1)C2)=O c1(CC(=O)NCC(C)N(C(=O)CC2CCC(C)O2)C)ccc2nn[nH]c2c1 CCC(C)C(C(=O)N1CCCC1(C(N1CC(C)(C(N)=O)C1)=O)CC)N(C)C C(=O)(CCCC(C)(C)NC(c1cn2c(n1)CCC2)=O)Nc1ccc(C)cc1O CN1CCC2CN(C(C3(C)CCCN(C(=O)CCc4ccc(Cl)s4)C3)=O)CC12 C1(C(=O)NC2CCC(C)(NC(=O)CN3CCOCC3)CC2)CC1C1CC(F)(F)C1 N1(C(CC2ON=C(C)C2)=O)CCOC(C(C)NC(C2CCCN(C(C)C)C2)=O)C1 C#CC1(O)CCN(C(=O)OC(C)(C)C)C1.N12C3CCC(C3)C1C(=O)N2 N1(C(C2(C)CC(C)(C)C2)=O)CC2CCCC(C1)N2C(=O)C(C)(C)n1cnnn1 Cn1nccc1CC(=O)NC(CNC(C1CC1C(F)(F)F)=O)C1CC1 CC(C)CC(O)C(=O)N(CC(C)(C)CNC(=O)Cn1ncc(C#N)c1N)C N1(C(CCN(CC)CC)=O)CCCC(C2CCN(C(=O)C(C)O)CC2)C1 CC1(C)C(CNC(=O)COC2CN(C(=O)C#CC3CC3)C2)CC1O N1(C(c2cncc(C)c2)=O)CCC2(CCCN2C(c2sccc2C2CC2)=O)C1 Cc1ccc(C(=O)NCC2COCCN2C(C2CC2c2ccc(O)cc2)=O)nc1 c1(C(=O)NCCC2CC(C)C2)cncc(CNC(C2(C)CNC(=O)C2)=O)c1 c1(C(C)C(F)(F)F)cccc(NC(C2CCCN2Cc2cccs2)=O)c1 c1(C(N2CCC(CNC(c3c(CC)c[nH]n3)=O)C2)=O)ccc(SC(F)(F)F)cc1 c1(NC2(c3nnnn3C)CC(CC(C)C)C2)cccc(N=[N+]=[N-])c1 N1(C(c2ccc(=NC)[nH]c2)=O)CC2(CC(NC(=O)C(C)NS(=O)(=O)CC)CO2)C1 c1(SCCC(=O)NCC(C)(C2CC2)NC(C2COCCO2)=O)ccc(C#N)cc1 N1(C(CCCC#C)=O)CCC(NC(=O)CCC2CCCO2)C(CO)CC1 C1(C(N(CCCO)C)=O)(NC(=O)CC2C(C)(C)C2(C)C)CCN(C)C1 c1(C(N(C)CC2CCN(C(CC)=O)C2)=O)c(F)c(F)cc(F)c1F c1(C(=O)Nc2c(C)ccc(N)c2)cc2n(n1)CCN(C(=O)C(C)(C)C)C2 c1(OC)cc(F)cc(C(=O)NCC(CO)NC(C2CCCC(F)(F)C2)=O)c1N N1(C(C(CN(C)C)O)=O)CCCN(Cc2cn(C3CC3)nn2)CC1 C12CN(C(C)(C)C1)C(c1csnc1OC)C(=O)N2.C1(C(=O)OC)(CF)CC1 CCCC(F)C(=O)N1C(C(=O)NC(C)C(=O)OC)CCC1C(C)C N(C1CCCOc2c(F)cccc21)C(COC(c1c(OC)cc(C)cc1)=O)=O c1(C(N2CC3CCN(C(c4nc(Br)cs4)=O)CC3C2)=O)cc(Cl)cc2cc[nH]c12 c1(NC2C(NC(c3n(C(C)C)ccn3)=O)CCCC2)nc(Cl)nc2c1ncn2C c1(SCC)ccc(CC(N2CCOC(CCNC(c3cncnc3)=O)C2)=O)cc1 C(CC(C)C(=O)N1CCC(O)(CCNC(c2n[nH]cc2C2CCC2)=O)C1)OC C1(CCCNC(=O)CSC(F)(F)F)(CNC(C(C)OC2CCOC2)=O)CCCC1 C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NCCCNC(CCC(CC)OC)=O C1(NC(c2c(CC)scc2)=O)CN(C(=O)C(C)(C)c2ccns2)CC1C CC1CN(C(C2CCC(=O)O2)=O)CC2(CCN(C(=O)C(C)(C)C(C)(C)O)CC2)O1 N1(C(C2C(=C)C2)=O)CC(OC)CC1CNC(c1ccc(OC)nc1)=O C1(CC(=O)NCC2(CCNC(C3(CC#C)CCCO3)=O)CC2)COCC(C)O1 C(N=c1ccn2c(Br)cnc2[nH]1)C1N(C(=O)CC2CC(F)(F)C2)CCCC1 CC(C)CC(C(=O)NC1CCOC1)ONC(c1cnn(C(F)F)c1)=O N1(C(C(CC)CC2CCCC2)=O)CC2CCC1CN2C(=O)C(C)(C)C(C)O CC(C)C(F)(F)CNC(=O)CONC(=O)Oc1ncn(C)n1 C(=O)(CCCC(CC)NC(=O)C(F)C(C)(C)O)N(C)Cc1cn(CC)nc1 C(=O)(CC(C(F)F)c1ccc(F)cc1Cl)N(CCNC(c1n(CC)ncc1)=O)C c1(C(N2CC(C3(NC(Cc4cncc(N)c4)=O)CC3)C2)=O)ccc2cncn2c1 c1(C(C)NC(c2ccc(C)cc2)=O)ccc2c(c1)COC2.C12CCCN(C1)C2=O N1(C(C2CCCN(c3nc(C)cc(C)n3)C2)=O)CCC2(NC(=O)CO)CCCC12 c1(C(=O)NC2CCC2(Cl)Cl)cccnc1NC(C1CC(SCCO)C1)=O.C1CO1 C1(CNC(CCN(c2ccc(C(=O)NC)o2)CC#C)=O)CC2(CC2)C1 N1(C(C(=O)N(C2CC(OC)C2)C)C2CC(SC)C2)CC(CC2CC2)OCC1C C(=O)(CCCc1ccccn1)NCCC(C)N(C(CCOC(C)C)=O)C c1(C(N(C2CCC(NC(C3CCCSS3)=O)CC2)C)=O)cccc2c1OCO2 N1(C(C2C(COC)C2)=O)CC2(CCC(CNC(c3nc(C)c(C)[nH]c3=O)=O)O2)C1 N1(C(C2C(C)(C)COC2)=O)CC2CC(NC(=O)CCOC3CCOCC3)CC1C2 CC1OC2(CO)CC1(NC(=O)C(=O)NC1CCOCC1F)C2 C1(C(N2CC(NC(c3cn(C(C)C)nn3)=O)C(C)C2)=O)CN=C2N=CNN2C1 CS(=O)(=O)c1ncc(C(N2CC3CC3(NC(=O)COC(F)F)C2)=O)s1 c1(C(=O)NC2C(NC(=O)C(=O)NC3CC3)CCC2)ccc(C(F)(F)F)nc1 CCCC(CC)CC(=O)N(C1CCN(C(c2ocnc2C)=O)C1)CC C1(NC(C2(CC#C)CCOCC2)=O)CCN(C(=O)C=Cc2ccccc2)C(C)C1 c1(C(C(=O)Nc2cccc(C(C)F)c2)NC(C2CC2(Cl)Cl)=O)c(C)cccc1Br N1(C(c2cc(CCC)oc2C)=O)CCC(NC(=O)CC2(C)OCCO2)C(CC)C1 N1(C(C2=NOC(CNC(=O)CC3CC4(CC4)CO3)C2)=O)CCCC2(CC1)CC2 C1(C(=O)NC2CC(CNC(c3ccc(C(N)=O)[nH]3)=O)C2)CCc2nncn2C1 C(CCCC(=O)NCC(O)C1(Cl)CC1)N(C(C1C(C(=O)OC)CC1)=O)C C(=O)(C1CCN(C)c2ccccc21)OCc1cncc(C)c1 C12(C(=O)NCCCN(C(c3c[nH]c(C)c3)=O)CC)CC1COC2(C)C C1(NC(C2CCN(C(c3cc(C)c(C)o3)=O)CC2)=O)CCN(C)CC1C#N C1(CCC)CN(C(=O)C(C)(C)CSC)CCN1C(=O)C(F)=CC1CC1 C(CC(C)(C)C(=O)NCC1CC1c1ccco1)NC(CC1(C)CCOCC1)=O C(=O)(C#CC(C)(C)C)NC(CNC(C1CCN(CC(C)C)C1)=O)(C)C1CC1 C(=O)(CC(C(F)(F)F)N(C)C)N1CCC(N2CCN(C(CCC=CC)=O)CC2)C1 N(C(=NCc1noc(C)n1)NC(C)Cc1ccccc1)C1C(C=C)C1 C1(C(=O)NCC2C(NC(c3ccn(CC)n3)=O)CC2)CCCC12CCC2 Cn1cncc1C=CC(=O)NC1CCCN(C(c2c[nH]nc2-c2ccoc2)=O)C1 c1(OC(CC)(C)C)ccccc1C(=O)NC1CC1CNC(=O)C(C)(C)C N1(C(C2(CC)COC2)=O)CCSC(C(N2CCC(N3CCOCC3)CC2)=O)C1 c1(NC(CC2CC(=C)C2)=O)c(CC)cccc1CC.C12CCN(CC1)C2=O Cc1[nH]nc(C(=O)NC2CC(n3cc(C4CCCN(C)C4)nn3)C2)c1Br S(=O)(=O)(c1cc(C(F)F)ccc1NC(Cc1nccs1)CO)NCC(C)S(N)(=O)=O C(=O)(C#CC1CCCO1)NC1CC(O)(CNC(c2c(Cl)sc(C)c2C)=O)C1 C1(N(CC(=O)NCC(C)NC(=O)CNC(=O)C(F)(F)F)C)CCCCC1 N(C1CC(C)n2ncnc21)C(CN(C(=O)CCCCN=[N+]=[N-])CC)=O Cc1ncnc(O)c1-c1nc(C2CCOC2)nn1-c1ccnc(Br)c1 c1(C(=O)NCC(CCC)NC(C2CCS(=O)(=O)C2)=O)ccc2nn[nH]c2n1 Cc1cccc(C2(CNC(=NCc3ccccn3)NCC3CCCC3)CC2)c1C N1(C(c2ccc(C)s2)=O)CC2CC1CN(C(=O)Cc1cccnc1)C2 C1(CC)COCC1NC(C1CCC(NC(C2CC(C)C2)=O)C1)=O C(C#Cc1ccccc1Cl)N1CC(C(C)NC(=O)C2=C(Cl)CC2)OCC1 c1(C(N2CC=CC(NC(c3oc(C)c(CO)c3)=O)C2)=O)ccc2cccnn12 Cc1cc(F)c(C(N2CCCC(NC(c3ccc(O)cc3C)=O)CC2)=O)c(Br)c1 c1(C(CC)NC(CC)C(=O)OCc2ccccc2)cc(Cl)ccc1F c1(C(N2CC3N(C(CCC(=C)Br)=O)C(CC3)C2)=O)nn(C)c2ccccc12 c1(C(=O)NCC2CCN2C(=O)C(O)CC2CCCCC2)nc2cccnc2s1 CC(CNC(C1CC1C(F)(F)F)=O)CC(=O)NC1CCNC(=O)C1 C1(CNC(c2scc(OC)c2)=O)CCN(C(=O)Cn2cnnc2O)CC1(F)F N1(C(=O)NC2C(C)C2)CCSC(C(F)(F)F)C1 Cc1cc(NC(C2(F)CC=CCC2)=O)cc(C(C)C)c1 N1(C(c2ccc(C#C)o2)=O)CCCC(C(=O)NC2CC(=O)N(CC)C2)C1C C12(NC(CN(CCC)C)=O)CCCC(CN(C(c3ccc(C(N)=O)o3)=O)C1)C2 C1(CC)CN(C(C2CCSC2)=O)CCN1C(=O)C(C)CC1CCCC1 c1(C(CNC(N(C2CCCN2C(N)=O)C)=O)(C)C)ccc(C(F)(F)F)cc1 c1(CN(C(=O)Nc2scc(COC)n2)C)c[nH]c2ccc(F)cc12 N1(C(c2c(OC)cc(O)nc2)=O)CC2CCCC1(CNC(=O)C(F)OC)C2 C1(C(=O)NCC(CNC(C2(C(C)C)CNC(=O)C2)=O)(C)C)CC(C2CC2)=NO1 c1(-c2ncc(C(c3nnnn3C3CC3)NC(CC=C)(C)C)s2)ccc(F)cc1 N1(CC(=O)NCC2CN(C(C(CCC)O)=O)CC2O)OC(C)(C)CC1=O C1(CCC(=O)NC(CC#C)CC)CCCN(C(=O)C(C)(C2(C)CC2)OC)C1 C1(C#N)(C(=O)NCCn2cc(C(=O)NCCN(C)C3CC3)nn2)CCCO1 c1(OCC(Cn2cc(CC(O)C3CC3)nn2)OC)snnc1C(=O)OC(C)(C)C N1(C(C(C)OCC(C)C)=O)CCCC12CCCN(C(=O)C1=C(Cl)CCCC1)C2 C1(C(N(CCCCNC(C2C(C)OCCC2)=O)C)=O)C(F)(F)C12CCC2 CCCCC(CC)CC(=O)NCc1ccoc1C(=O)N(C)CCN1CCCC1=O C(CCC(F)(F)F)(c1ccccc1)N.CC1CCCN(C(C)C(=O)O)C1 C(=O)(CC(C)(C)CN(C)C)NC(CNC(c1ccc(SC)s1)=O)(C)C1CC1 c1(C(=O)NC2CC(NC(CN(CC)CC)=O)C2)cc(O)ccc1Cl c1(OC)ccc(C(N2CCC(CNC(C3CCO3)=O)CC2)=O)nc1 N1(C(=O)CCCC2CCCO2)CCN(C(C23CCC(CC2F)C3)=O)C2(CC2)C1 C(N=c1ccnc(CNC(c2nn(C)c(OC)c2C)C)[nH]1)C1(CCC)CCC1 C1(CC(=O)NCCn2ccc(C(=O)NC34CCCC3C4)c2)NC(=O)NC1=O C1(C(=O)NCC2C(=C)C2)(OC)CCN(C(=O)CCNC(c2ccco2)=O)C1 C#CCCCCC(=O)NCC1CCC1NC(c1ncoc1-c1ccccc1Cl)=O c1(NC(=O)NC(C(=O)N(CC(=O)OC)C)(C)C)ccc2cnccc2c1 C(CC(C)S(C)(=O)=O)N(C(C)(C)C)C(=O)NCc1cccc(C(=O)NC)c1 c1(CC(=O)NC2CC(CNC(C(C)N(S(C)(=O)=O)C)=O)C2)cn2c(n1)CCCC2 N1(C(C2N(C(C34CC(C#N)(C3)C4)=O)CC3CCCC32)=O)CC2C3CCC(O3)C2C1 C(=O)(C(CCN(C)C)N(C)C)N(C(CNC(c1scc(C(=O)OC)c1)=O)C)C C1(C)(CC)C=C(C(=O)NCC#CCNC(c2ccc(OC)cc2OC(C)C)=O)C1 C12(NC(c3cccnc3O)=O)CCCN(C(C3CCOCC3)=O)CC1C2 c1(C(=O)NC(CN(C(=O)CN2CC(C)C2)CC)C)cnn2ccc(Cl)c(F)c12 C1(C(=O)NC2C(NC(C)=O)C2)CC2C=CC1CCC2 n1(CC(=O)NCCC2N(C(C(C)(O)C3CCC3)=O)CCCC2)cnc([N+](=O)[O-])n1 N1(C(C(C)N(CC)CC)=O)CCn2ncc(CNC(=O)CC3CCC(O)C3)c2C1 C1(C(=O)NCCC(=C)CNC(=O)CCN2CCCCC2=O)CCCC(C#N)C1 C1(NC(Cc2c(C)n(C)cn2)=O)CC12CCN(C(=O)C1=COCCC1)CC2 c1(C(=O)NC2CCN(C(CSC)=O)C(C3CC3)C2)c2c(nn1C)CCSC2 c1(C(N2CCC(C)(NC(=O)C(c3ccccc3)F)C2)=O)cccn2ncnc12 c1(CNC(C(n2c(C)ncc2)C)=O)ncccc1C(=O)N(CCO)CC1CC1 CC(C)CC(C(=O)NC1CC(C)(C)C12CC2)NC(c1cccc(O)n1)=O C1(C(N(CCNC(=O)CC2CCCC2)CC)=O)CC2CC1CC2(F)F CC(C)C(F)(CNC(C1CCN(C)C(=O)C1)=O)C(=O)NCCC1(C)CCOCC1 C(=O)(CS(N)(=O)=O)NC1(c2ccccc2)CN(C(C2(N(C)C)CCOC2)=O)C1 N1(C(C(C=C)OC)=O)CCC(O)CC1C(=O)NCC1(C2CC2)CC1 C(CCC(C)(C)C(=O)N1CC(C)=C(C)C1)NC(C1CN(CCC)C(=O)C1)=O c1(C(=O)NC(CNC(C(CC)(CC)CC)=O)(C)C(C)C)cn2c(n1)CCC(C)C2 Cc1n[nH]c(C)c1C1CC(Nc2ccnc(O)n2)CCO1 C1(CNC(c2c(CC)nc[nH]2)=O)CC2(CCC2)CN1C(C1CC1[N+](=O)[O-])=O C(C)(CC(=O)NCC(C)(CO)NC(=O)COC(C)C)=CC N1(C(c2c(CC#N)ccs2)=O)CC(NC(C2(C)CCCO2)=O)C2CCCCC12 C(=O)(CC(C(F)(F)F)NC(C1(CC(C)C)CC1)=O)NCC(C(=O)NC)O C1(C(=O)NCC2(F)CC(CNC(C(CC)O)=O)C2)CCCCN1C1CCCC1 C1(CCC(N2CCC(C3C=NC(O)=[N+]3F)C2)=O)CCCN(C(=O)CCOC2COC2)C1 C(C(CC1CC1)C(=O)NC(C)(C)C(N)=O)NC(COCCCOC)=O C1(CC)C(C(=O)NCCSC)CCN1C(=O)CN1CCSCC1 N1(C(c2c(CC)con2)=O)CC=C(C(=O)NCC(C)(COC)CO)C1 CCCC(C)(CC)C(=O)NCC1CCN(C(c2cc(C)no2)=O)C(C)C1 C(CC(C(=O)O)N(C(=O)CC1CC2CC2C1)C)SC c1(OC)cc(C)c(C(=O)NCC=CCNC(C2CCCC(F)C2)=O)c(C)c1 C(=O)(C(C(C)C)C(C)C)NCC(CCC)NC(C1(Cl)CC1)=O C(CC(C(=O)NCC(C)C(C)(F)F)NC(c1cccc(CO)n1)=O)SC N1(C(C2CCN(CC)C2)=O)CCCCC(C(=O)NCCCC(C)C)C1 N1(C(C2(CC)CCCO2)=O)CCCC(CCC(=O)NCC(C)OC(F)F)C1 N1(C(C(C)CC2CCCO2)=O)CC(C2CN(C(c3ccccc3Cl)=O)C2)C1 C1(C(=O)NCCCC2OCCN(C(C(C)NC=O)=O)C2)CC(=O)NC(=O)N1 CC1CCCCN1CC(=O)NC(c1nocc1C(=O)Nc1c[nH]nc1C(N)=O)C C1(NC(C(CCSC)O)=O)CN(C(=O)CC2CCS(=O)(=O)CC2)CCC1O c1(C(=O)NC2CN(C(CCC(C)C)=O)C(C)CC2)cnc2c(F)cccc2c1 C(C(C)(C)CC(C)C)NC(C1(CF)CCN(C(CCC(C)C)=O)C1)=O c1(C(C)NC(=O)C(=O)NCCc2cccc([N+](=O)[O-])c2)ccc2oc(O)nc2c1 c1(CC(C)C(N2CCC(C)(NC(c3cc[nH]c3)=O)C2)=O)ccc(Cl)cc1 C1(CNC(C(CC)NC(C)=O)=O)C2CN(C(=O)CCn3ccnc3)CC12 C(C(C(C)C)NC(C1(C)CN(c2ccccc2)C1)=O)NC(C(F)=CCC)=O N1(C(C2CCC(NC(=O)CCc3cscn3)C2)=O)CCCc2occc2C1 CC1C(NC(=O)Cc2ccn(C(F)F)n2)CCCN1C(c1ccc(Cl)[nH]1)=O N1(C(CCCOCCC)=O)CC2CCCC2(C(N2CC(C)C2(C)C)=O)C1 C1(NC(c2cc(F)c[nH]2)=O)CCN(C(c2ccc(CO)cc2)=O)CC1 CC1=NN(C)C(=O)C1CC(N1CC(C)C1CNC(=O)CC12CCC(CC1)C2)=O S(=O)(=O)(c1c[nH]ccc1=NC1CCCC(C)C1)NC(CC)CC C(N=C(NCC1(C)CCCCC1)NC1CC1)C1C(C)C1 N1(CC)CCCN(C(=O)C(C2CCCO2)OC)CC1.c12nccn1C2 CCC(C)(C)CCNC(C1CCN(C(=O)C(C)c2ccco2)CC1)=O C(=O)(NNC(=O)C(N)C(C)(C)C)c1ccc(OC)c(Cl)c1 S1(=O)(=O)c2ccc(cc2)C(=O)N(CCC)CCCN1.C(=O)(C(C)=CC)NC(C)C c1(C(N(CC(=O)NC2CN(C(C)C)C(=O)C2)C)=O)ccn2ccnc2c1 c1(C(=O)NCC2N(C(C3C(=O)NCC3)=O)CCC2)cc2c(Cl)nccc2o1 Cn1cc(C2(C(=O)NCC3CCCC3NC(=O)CC3CC34CC4)CCCO2)cn1 N1(C(c2ccc(CC)nc2)=O)CC(NC(c2cc(Br)c(C)o2)=O)CC(O)C1 C1(C)C(CC(=O)N(c2c[nH]c(=N)c(C)c2)C)NC(=O)N1.Cc1ncsc1CO C1(NC(C2CC(C)(C)OCC2)=O)CC2CC(C1)N(C(C1C=CC=CC=C1)=O)C2 C1(CC#N)CN(C(c2cc(O)nc(O)c2)=O)CCN1C(c1cc(Cl)cs1)=O C1(C(=O)NC2CCC(NC(c3c(C)cno3)=O)C2)COc2ccccc2C1 N1(C(CC)=O)CCCC2CN(C(c3ccc(OC)cc3O)=O)CC12 C=CCC(C)(CC)C(=O)NCC1C=CCN1C(c1ccc(Cl)cc1F)=O c1(C(=O)NCC2(C)N(C(C=CC=CC)=O)CCC2)ccc2c(c1)nc(O)n2CC N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC2(C1)CN(C(C1CC3CC1C3)=O)CCO2 c12ccccc1CN(C)C2C(=O)Nc1csc(C2CC2)n1.C1(CCC)CCCCC1 c1(C(N(C2CCCN(C(=O)C(O)CF)C2)CC)=O)[nH]nc([N+](=O)[O-])c1Cl c1(C(N)=O)nc(C(=O)NCCCCCNC(=O)CCc2ccncc2)cs1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(NC(c2csc(C3CC3)n2)=O)C(O)C1 N1(C(CN2CCC(N(C)C)CC2)=O)CCC(n2cc(C3(O)CSC3)nn2)C(O)C1 C1(NC(CC2(C)CC2(Cl)Cl)=O)CN(C(c2ncccn2)=O)Cc2nccn2C1 c1(OC)cccc2c1CCC2NC(c1nnnn1C(C)C)C.c12ncc(s1)C2 Cc1cc(C(=O)NCC(C)CC(=O)N2CC(C)(F)C2)c(C)[nH]1 S(=O)(=O)(c1ccc([N+](=O)[O-])c(F)c1)N(CCC(N1CCC2CCOCC2C1)=O)C C1(C)(C(=O)NCC2(CC)CC(C)(C)C2)CN(C(C2CC(C)(C)C2)=O)CC1C CC1(NC(=O)CCCC2CCC2)CC(NC(=O)C(C)(C)c2cccnc2)C1 C1(N(C(C2N(CC)CC2)=O)CC)CCCN(C(=O)C(C)O)C1 c1(C(=O)NC2C(CNC(CS(=O)(=O)NCC)=O)CC2)cnn2c1OCC(C)C2 N1(C(c2[nH]cc(C)c2C)=O)CC2(CO)CC1(C(=O)NC(C)CC1CCC1)C2 C1(NC(c2cc3oc(Cl)cc3[nH]2)=O)CCC2CN(C(=O)CCC3CCC3)CC2C1 CCCCCC(C)CC(=O)NCC(C)(CO)NC(=O)C(c1cccn1C)=O Cc1cc(C(=O)NC2COC3(C2)CN(C(=O)CC2(C)CCCO2)C3)c(O)nc1C C(=O)(C(C)CCC)N(C1CCCC1)CCCNC(c1nc(CCC)sc1)=O CC1C(C(=O)N2CC3(CCCC3)C2C(N2CCCC3(C2)N=N3)=O)=NOC1C N(C1CCCc2c1cnn2C1CC1)C(C)=O.C1CCC(C(N(C2CC2)CC)=O)CC1 Cc1cc(C(N2CCC(F)C(NC(=O)COc3ccon3)C2)=O)cc(C)c1 CS(=O)(=O)c1cc(C(N2CC3CC(CNC(c4ccc(Cl)o4)=O)CC2C3)=O)co1 c1(C(=O)NCc2c(C(C)C)ocn2)cn(Cn2cc(C(O)C(C)C)nn2)c(C)n1 C1(O)(CN(C(C2C(CC)C2)=O)C)CN(C(c2ccsc2C)=O)C1 N1(C(C(CCC)OC)=O)CC(NC(=O)CSCC(F)(F)F)CC12CCCC2.C(C)(=O)N N1(C(c2c(CC)ncs2)=O)CCC(C)(C)C1C(N1CCC(Cn2ccnc2)CC1)=O c1(C(=O)NCC(CCCC)NC(C)=O)ccc2c(c1)C(=O)N(C)C2=O n1(CCC)nccc1CNC(c1cnc(C2CCCO2)s1)c1nnnn1C c1(CC)cc(C(N2CC(NC(=O)C(C)(C)O)C(F)C2)=O)ccc1Cl N1(C(=O)OCC2N(C(CCCCC)=O)CCCC2)CCCC2(C1)NC(=O)NC2=O C1(NC(C2(NC(C3CC(F)C(=O)N3)=O)CSC2)=O)CC2(CCC2)C1 c1(COCCOCCNC(CC2CCC(C)(C)CC2)=O)ncc2cccnc2n1 C1(NC(=O)C=Cc2ccoc2)CC(C(=O)NC(CN(C)C)CO)CC1O C1(C)(NC(C(C)N(C)C)=O)CN(C(=O)C(C)(C)c2ncco2)C1 C1(CN(C)Cc2cc(C(=O)O)nn2C)CCN(C(=O)CC2CC2C2CC2)CC1 C1(C(=O)NC2CCN(C(c3c(CSCC)cccc3)=O)C2)CN2CCN1CC2 C1(CNC(C2CC2c2ccoc2)=O)C=CCN1C(=O)Cn1ccc(C2CC2)n1 C1(OC)CCC2(C(N3CC(F)(CNC(C4CC4Cl)=O)C3)=O)CC12 CCC(CC)C(=O)NC1CC(N(C(=O)C(c2ccccc2)=CC2CCCO2)C)C1 C1(c2n(C(C)(C)C)nnn2)(Nc2cccc(O)c2)CCC2(CCCOC2)C1 C(c1ccccc1Cl)=CC(=O)NCC1(F)CCC(NC(COCCCC)=O)C1 C=CCC(C)C(=O)N1CC2CC2(CNC(=O)C(C)(C)CF)C1 CS(=O)(=O)CC(=O)NCC(O)CNC(=O)CC1(Sc2cccnc2)CCCC1 C(C(C(C)(C)C)NC(=O)CNC(C1CCC1)=O)NC(C1C(=C)CC1)=O c1(C(N2CC3CC3(C(=O)Nc3cnc[nH]3)C2)=O)ccc(Cl)cc1Cl c1(C(N)=O)cccc(C(=O)NC2CC(NC(c3ccc(C(F)F)cc3)=O)C2)c1F C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(c2cc3ncccc3s2)=O)CCC1(C)C CC1CCC(C(=O)N(CC(C)O)CCNC(c2csc(Br)c2)=O)CC1 N1(CC(=O)N(CC(CC)NC(=O)C(C)n2cccn2)C)CCNC(=O)C1 c1(C(C)=O)cc(Br)c(C(=O)NC2(CNC(=O)CC3CCCCO3)CC2)s1 C1(NC(C=Cc2ccc(SC)cc2)=O)CC2CCC1N(C(=O)C(C)S(N)(=O)=O)C2 c1(NC(C2(C)CCN(C(CCOC)=O)C2)=O)cccc(C)c1C(F)(F)F C#Cc1cccc(C(N2CCOCC(C(=O)N(CC(O)COC)C)C2)=O)c1 NS(=O)(=O)c1cccc(C(=O)NCC2CCCCN2C(C2(CCO)CC2)=O)c1 Cc1ncc([N+](=O)[O-])c(N(C)CC2CN(C(C3CCc4n[nH]cc4C3)=O)C2)n1 c1(C(C)NC(c2cc(CC)c(OCC(=O)OC)cc2)=O)ccc(Cl)c(C)c1OC C1(N(C)C(c2occc2Cl)=O)CC2CCC(C1)N2C(C1CCn2ncnc2C1)=O N1(C(c2occc2CC)=O)CCCN(C=O)CC1.C1(CCC)(COC)CCNC1=O Cc1cc(C(=O)N(C2CN(C(=O)CCCc3cnccn3)CC2F)C)c(C)cn1 C1(C(=O)NC2CCC(NC(c3c[nH]c(Br)c3)=O)C2)(COC)CCC(=O)N1 Cc1nc(C(=O)NC2CC(NC(C3CCC(=O)NC3)=O)C2)nn1C c1(C(N2CC(C)(NC(C3C(C=C)OCCC3)=O)C2)=O)ccc(C)c2cccnc12 Cn1cc2c(C(N3CCC4(C3)CN(C(=O)C(F)F)C4)=O)cc(F)cc2n1 C1(NC(C2(OC)CC2)=O)C2CCN(C(=O)C(C)CC3CCCC3)CC12 C1(NC(CCc2n(C)ncc2)=O)CCC2CC1CN2C(c1occc1Cl)=O C1(NC(=O)C#CC2CC2)CCCCC1N=c1[nH]c2cc(F)ccc2o1 CCC(C(=O)NCCN(C(C1CC1C(F)(F)F)=O)C(C)C)SC CN1CC(C)(C)CC1C(=O)NC1(CO)CCCN(C(c2ccoc2)=O)C1 CC(C)CC(CNC(c1ccnnc1)=O)C(=O)NC1CCCC12CC2 C1(C(N2CCN(C(C(c3c(C)cccc3)C)=O)CC2)=O)Cc2c(F)cccc2O1 c1(CNC(C2CCC(COC)C2)=O)ccc2c(c1)CN(C(=O)CCOC(C)=O)C2 C=CCCCC(C(=O)Nc1cc(C)cnc1OC)NC(=O)C(F)C(C)(F)F C(CN=c1ccc(S(=O)(=O)N2CCN(C)C(CO)C2)c[nH]1)C1CCN(C)C1 C1(C(N(CCCCNC(=O)CN2CCCC2)C)=O)(CC2CC2)CCOCC1 C1(C(N2CCCC(NC(c3n(C(C)C)ccn3)=O)C2)=O)CCCC12CCOCC2 c1(C(=O)NC(C2CCN(c3ncccn3)C2)C)cccc(P(C)(C)=O)c1 C1(C(C)NC(CC(n2ccc(C)n2)C)=O)CCCN(C(=O)CNC=O)C1 N1(C(C2(CC)CCCCC2)=O)CCC2(C1)CN(C(=O)CSC(C)(C)C)C2 Cn1ncc(C(=O)Nc2ccc(O)cc2)c1C(F)F S(=O)(=O)(c1ccc2[nH]c(=NC3CCN(CCF)C3)sc2c1)NC1C(C)(C)COC1 c1(N(C(c2c(C)cccc2Cl)=O)CC2CNC2)ncc2c(n1)NC(=O)C2 C1(NC(N(CCC(C)C)Cc2ccsc2)=O)CCC(c2ccccc2)O1 C1(CCC)CN(C(=O)C(C)S(N)(=O)=O)CCN1C(c1sc(C)nc1C)=O Cc1cccc(C(=O)NC2CCCC2NC(C2(C3CCCCO3)CCC2)=O)c1F c1(C(=O)NCC2(C(N)=O)CN(C(C3(C=C)CCC3)=O)C2)cc(Cl)nnc1O C1(NC(C(CC=C)N(C)C)=O)CCC12CCN(C(=O)CC(C)F)CC2 C(=O)(CCCC(CCC(=O)OC)NC(=O)NCC1CCCC(CO)C1)OC C1(C(=O)NC(c2cccnc2N)C)CC1C1CN(C(=O)OC(C)(C)C)C1 C#Cc1cccc(C(=O)NCC(CC=C)C(=O)N2CCC(SC)CC2)c1 c1(CSC(c2cnc(C(F)(F)F)o2)C)ccncc1Cl C#Cc1ccc(-c2nc(C(=O)NCCN(C)CCO)cs2)c(C)c1 C(=O)(C1CCc2ccc(OC)cc21)NCC.CCCC(C)C(=O)NC CC1(C)CC(CNC(c2ccc(OCC(F)(F)F)o2)=O)CN1C(=O)C1=CCOC1 N1(C(CCSCCCC)=O)CC(NC(=O)CN(C)C(c2ccsc2)=O)CC(C)C1 c1(C(=O)NC2C(CNC(C3CC(OCC)C3)=O)C2)ccc(F)cc1Br C1(CCNC(CC=C)=O)CCCN(C(C2CCC(=O)N2c2cnccn2)=O)C1 c1(C(=O)Nc2cncc(C(F)C(F)(F)F)c2)ccc2ccc(O)cc2c1 C(=O)(C1=CC2CCCC12)N1C(CNC(C2(C)CCN(C(C)=O)C2)=O)CCC1 c1(NC(C(=O)NCC2CN(CC)C(=O)C2)=O)ncc(C#N)cc1C c1(NCC(N2CC(C(C)NC(C3(C)C(CC)CCC3)=O)C2)=O)cccc(C#N)c1 c1(C(=O)NCC2CCN(C(C(CSC)C)=O)C2)cc(C)c2c(O)n[nH]c2n1 c12ccc(cc1)C(=O)NC2.C1(CN(C)C)CCCO1 c1(C(=O)NC(C)C(CO)NC(C2CNC(=O)C2)=O)nc(Br)c2ccccn12 c1(OC)cn(C)c(C(=O)OCC(=O)NC(c2ccc(OC)cc2)C)cc1=O C1(CC(=O)NCCCC(C)NC(c2ccsc2Cl)=O)CC2CCC1O2 C1(C(=O)NC2CCN(c3ccc(C)nc3)CC2)Cc2c(ccc(F)c2F)CN1 c1(C(N2CCC(CNC(C=C(C)Cl)=O)C23CCC3)=O)cc2ccccc2nc1O C(=O)(C#Cc1ccccc1)N1C(C(=O)Nc2c(CC)nccn2)CC(F)C1 CC1C(NC(C2C3CCCC23)=O)CCN1C(C1(n2ccnc2)CCCC1)=O C(=O)(CCCNC(c1cnc(OCC)s1)=O)NCCCOCCOC c1(C(=O)NC(CC)C(=O)NC(c2nccc(O)n2)C)c(C)cccc1C N1(C(c2c(C)n(CCN(C)C)cc2)=O)CCCC2(C1)CN(C(c1ccsn1)=O)C2 c1(C(=O)NCC2C(OCC)CN(C(C3CC(C#N)C3)=O)C2)cc(Cl)ccc1C C(=O)(C(CO)C(C)(C)C)NCCOCCNC(Cc1c(C)scc1)=O C(=O)(C1=CCCCCC1)NC(C)(CNC(C1CC2CCC1O2)=O)C1CCC1 C=CC(CCC)CC(=O)NC1C2CCC1N(C(c1ccn(C(C)C)c(=O)c1)=O)C2 CCCCCC(C)(CC)C(=O)N1CC(OCC)C(CNC(C2(C)CCOC2)=O)C1 C(CC(F)(F)CO)n1cc(C(C)N(c2cnn(C)c2)C(C2CC=CCO2)=O)nn1 C1(NC(=O)CCNC(=O)COC2CCC2)(CSC2CCOC2=O)CCCC1 N1(C(c2cnn(CC)c2Cl)=O)CCC(O)C(NC(=O)Cc2nonc2C)C1 N1(C(C2N(C(C3CCCO3)=O)CC(=O)NC2)=O)CCCC2(CCCC2)C1 CC(C)CCC(F)C(=O)N1CCCCC1C(=O)NC(CCl)C(F)(F)F N1(C(c2cccc(CC)n2)=O)CCN(C(C2SCC=C2C)=O)CC1CCO CCCS(=O)(=O)C(C)C(=O)NC1CCC1CNC(c1ccc2c(c1)OCC2)=O N1(C(CC#N)=O)CCC(NC(C2CCCSC2)=O)CC1 C1(OCCCNC(=N)N)CC2CCCC2N1C(C12C3C4C5C3C1C5C24)=O Nc1cccc(Cl)c1C(=O)NC1CC1NC(c1ncoc1C1CC1)=O c1(C(N2CC(N(C)C(c3ccn(C(C)(C)C)n3)=O)C2)=O)nccnc1N N1(C(CCCCCC)=O)CCC=C(C(=O)N2CC3(C2)CC3(F)F)C1 c1(C(N2C(C(N3CC(CC(=O)OC)C3)=O)CC(O)CC2)=O)cccc2c1CCC2 C12(CNC(=O)Cn3cccn3)CC(C1)C(NC(=O)C(F)(F)C1CC1)CO2 CC1(C)CCCN(C(C2CC3(CC(NC(C4(CCCF)CC4)=O)C3)C2)=O)C1 C1(NC(COC(CC)C)=O)COCCN(C(=O)C(F)(F)c2ccccn2)C1 c1(OC)cc(C(=O)NCC(C2CCOC2)NC(=O)CCC=CC(C)C)ncn1 c1(C(=O)NCC2(C)CCN(C(C3(COCC)CC3)=O)C2)cnn(C)c1C(C)=O C(=O)(CC(C)(C(F)F)N(C)C)NC1CCC(NC(c2c(C)cc(F)s2)=O)C1 Cc1cc([N+](=O)[O-])ccc1N1CC2(CN(C(c3cc(CC4CC4)on3)=O)C2)C1 C(=O)(CC1CC(=O)Nc2ccccc21)NC1C2CN(C(CC=CC)=O)C1C2 C1(C(N2C(CNC(=O)Cc3ccon3)CCC2)=O)CC12CCOC2 N1(C(C(C)NC(N)=O)=O)CCC(NC(c2cc(F)cnc2O)=O)C(O)C1 N1(C(C2(OC)CC(C(F)(F)F)C2)=O)CCC(NC(=O)C(C)C)C12CCC2 N1(C(C(C)OCCOC)=O)CC2CCCC(N(C(=O)CC(C)C(F)(F)F)C)C2C1 N1(C(CC2C(C)CC2)=O)CC2CC(C)N(C(=O)Cc3c(Cl)cccc3Cl)C2C1 c1(C(=O)NC(=O)CN(CCO)CCCC(F)(F)F)cccc2cccnc12 c1(OC)ccc(C(N2CC(O)(CNC(C3CC34CCC4)=O)C2)=O)c(O)c1 C1(CNC(C2C(C(C)C)CCC2)=O)CCC2(CN(C(c3cc(N)ccn3)=O)C2)O1 N1(C(CCN(C(C(C)C)=O)C)=O)CCCC(CNC(=O)COC2COC2)CC1 C(=O)(C(CNC(c1ccc(C)c(O)c1)=O)C(C)(C)C)NC1C(CC=C)COC1 CCCCC(F)C(=O)N1CCN(C(c2cccc(C=C)c2)=O)C(CC)C1 C=C(C)c1cn(CC2C=CCN2C(=O)CC2CC2(Cl)Cl)nn1 N1(C(CCN2CCN(C)CC2)=O)CC2(CC2)CC1C(=O)NCC(C)(C)O N1(C(C(n2ccc(C)n2)C)=O)CCC2(CC(C(NCP(C)(C)=O)=O)C2)C1 C=C1CCC(C(=O)NCC2CC(F)CN2C(C2CCCN2CCC(C)C)=O)CC1 CCC(C)CC(C(=O)N1CC(F)(F)CC1C)NC(C1C2CCCC12)=O Cn1cc(NC(C)(C)C2CC2)cc1C=O.c1(OCc2cccs2)ccc(OC)nc1 CC(c1ccc(F)cc1)=CC(=O)N(C1CN(C(=O)CCn2cccn2)C1)C C(C(C(C)C(C)C)NC(C12CCC(CC1)CC2)=O)NC(CC1(COCC)CC1)=O c1(-c2cc(CC(N3CC(COC)N(C)CC3)=O)ncc2)ccc2[nH][nH]c(=N)c2c1 C(CCO)(C(=O)NCC(O)CNC(=O)Cn1ccc(Br)n1)N(C)C C(=O)(C1CCc2c(Cl)cccc21)N1CCCC(NC(=O)C=CCO)C1 c1(C(=O)NCC(CN(C)C(C2CCCS2)=O)(C)C)cc(Cl)c(Cl)c(Cl)c1 CCC(C)CC(=O)NCC1CCCN(C(C2CCC(C(N)=O)CC2)=O)C1 c1(NC2(C)N(C(C#C)=O)CC2)nnc(-c2ccc(Cl)cc2)cc1C(=O)OC NS(=O)(=O)N1CCCC(C(N2CC3CC(C2)N(C(=O)CC2CS(=O)(=O)C2)C3)=O)C1 c1(CC)ccc2cc(C(=O)NC3CCC(N(C(=O)CC(C)F)C)CC3)ccc2c1 c1(C(=O)NCC2N(C(C(C(CC)C)N(C)C)=O)CC2)ccc2nc[nH]c2n1 c1(C(N2C(C(C)NC(C3CC4C=CC3C4)=O)CCC2)=O)ccc(O)cc1F Cc1cc(C(N2CC3CC3(CNC(=O)OC(C)(C)C)C2)=O)cnc1C(F)(F)F O(NC(=O)CN=c1nc(N2CCC(CC(=O)NC)CC2)c2sccc2[nH]1)CC CC(C(F)C(=O)NC1CC2(CCCN(C(=O)CC(C)(C)C(F)F)C2)C1)C(F)(F)F C1(NC(C2C(C)(C)C(F)(F)C2)=O)CC2CCC(C1)N2C(=O)CC1CC2(CCC2)CO1 c1(C(=O)NCCCN(C(=O)C(C)C(C)C)CC)ccnc2c1CCC2 c1(C(=O)NC(CCOC)C(=O)O)cn(C2CC2)c(C)cc1=O C1(NC2CCC(CC(=O)OCC)C2)CCCCCN1C(=O)OC(C)(C)C c1(C(=O)NC(CCNC(C(C)OCCC#C)=O)C)ccnn1CCCC C1(NC(c2ccc(C(F)F)nc2)=O)CCN(C(=O)C(F)=CC2CC2)CC1CO C(c1ccc(F)cc1)=C(C(=O)NCCOCCN(C(C1(F)C(C)C1)=O)C)C CC#CCCCC(=O)N1C(CNC(=O)CC(C)(C)OC)CC2CC12 c1(C(N2CC(O)(CNC(Cc3n(C)ncc3)=O)C2)=O)c(C(F)(F)F)cncc1F C1(CNC(c2cnn(C)n2)=O)CCCC2CN(C(C3CCC(Cl)CC3)=O)CC12 c1(CCC(=O)NCC(C)NC(C2CC2C2CCC2)=O)nc(O)c2ccccc2n1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C(=O)COC(F)F)CCC1C1CC1 c1(C(=O)NCCCN(CC)Cc2cncnc2)ccccc1CO C(=O)(CCS(=O)(=O)c1cc(Cl)ccc1Cl)OC(C1CC(F)(F)C1)C(=O)OC C1(CC(N)=O)(CNC(c2c(CC)c[nH]c2)=O)CCN(C(C2(CCO)CC2)=O)CC1 C1(C)(CC)CC(NC(C2(COC)CCOCC2)=O)CN1C(=O)CSC(F)F c1(OC)nc(C)cnc1C(N1CC(O)(CCNC(C2COC(=O)O2)=O)C1)=O c1(NC2C(SC)CCCC2)ncccc1S(=O)(=O)NC(C)C1=CCN(C)CC1 c1(C(=O)NC2CCCC(NC(=O)C=CCF)C2)cc2cc(C(F)(F)F)ccc2[nH]1 c1(NC(CCC)C(=O)N2CCCC(C)C2)ccc(-n2cccn2)c(C)c1 N1(C(C)C)N=C(C(=O)NCC2(C)CCN(C(C3CC(C)N(C)C3)=O)C2)CCC1=O N1(C(CC2C(CC)C2)=O)CC(N(C(=O)CCC2CC2(Cl)Cl)C)C(C)(C)C1 CC1CC(NC(=O)C(C)O)CN(C(=O)CCc2ccccc2O)C1 C(CCCCC(=O)NCC1(CO)CCC1)N(C(CC1C(C)OCC1)=O)C CCC(CC)C(=O)NCC1CN(C(c2ccc(N)cn2)=O)C2CC12 C1(CNC(=O)COCC2CCOC2)CCC(NC(C2CCCN(CC)C2)=O)CC1 C(=O)(C1=NOC(C)(C)C1)N1CCC(NC(c2cn(C(C)C)nc2)=O)C(O)C1 c1(C(N(CCCNC(=O)COC2CC=CC2)C)=O)cc(Cl)c(Br)cn1 C1(C(N(CCN(C(C)C)C(c2ccnn2CCF)=O)C)=O)CC2CC2C1 C(=O)(C(Cc1ccccc1)CC(C)C)NCCN(CCC)C(C12COCC1C2)=O N1(C(c2c(CCC)nco2)=O)CCC(C)(C)C(CNC(=O)C(C)C(C)C)C1 c1(C(=O)NCC(C)CNC(c2cccc(Cl)c2N)=O)coc2c(F)cc(Cl)cc12 Cc1cc(N(C)CCN(C(=O)C=CCCc2ccccc2)C(C)C)cc(C)c1 c1(C(=O)NC2CCN(C(c3scc(OC)c3)=O)CC2F)cn2cc(C)ccc2n1 c1(N2CCN(CC)C(C)(C)C2)nc2cc[nH]c2c(=NCc2c(C)noc2C)[nH]1 c1(C(N2CC(N(C(CC(C)C(F)(F)F)=O)C)C2)=O)cc2n(c1)CCS(=O)(=O)C2 Cc1c(C(=O)NCC2(O)CN(C(=O)C(c3ccc(F)cc3)=O)C2)cnn1C1CC1 C(=O)(C1=CCOCC1)N1CCC(CN(C(C(CC)NC(C)=O)=O)C)CC1 c1(C(=O)NC2CN(C(CC(C=C)(C)C)=O)CC(C)C2)cccc2c1CCOC2 c1(CC(=O)NC23CCC(NC(CC(C)CF)=O)(CC2)C3)ccc(S(N)(=O)=O)cc1 c1(C(=O)NC2CC(CCNC(C=NOC)=O)C2)c[nH]c2ncn(C(C)C)c12 N1(SCCOC)CCN(C(=O)Nc2ccc(CSC3CCCC3)cc2)CC1 c1(C(=O)NC2CCC3(CC2)CC3)ncnc(N2CC3C(NCC)C3C2)c1F C=CCC(CC)N=c1nc(N2CCC(c3cnccn3)C2)c2sccc2[nH]1 c1(-c2nnc(C)o2)nnc2n1C(C)CN(C(c1ccc3cc1NCCC3C)=O)C2 N1(c2cc(CC)ncn2)C2CCC1CC(CNC(=O)CCc1c(C)noc1C)C2 c1(CN(C)CCOc2ccc(C(F)(F)F)cc2)ccc2sccc2c1 C1(C(C)NC(c2cc[nH]n2)=O)CCN(C(=O)COCC2CCCOC2)CC1 N1(C(c2c(C)nccc2Cl)=O)CC2(C1)SCCC2NC(=O)CCc1ccccc1 C1(NC(C2CCCC2)=O)CC1C1CCN(C(c2cccc3c2OCO3)=O)CC1 C12(C(=O)NCC(CCNC(CC(n3ccc(C)n3)C)=O)O)CCCN(CCC1)C2 CCC(CCCC(=O)Nc1ccc(N)c(C)c1C)NC(=O)CS(=O)(=O)NC C#CC(C)(C)C(=O)NCC(C1CCCN(C(c2sc(CC)nc2C)=O)C1)(C)O C=C(C)CCC(=O)N1CCCC(N(C(=O)CCc2conc2C)CCO)C1 N1(c2nnc(CCOC)s2)CCC2(CCCC2NC(=O)COC2CCOC2)CC1 c1(C(=O)NCC2CCN(C(C3N(CC)CCCC3)=O)C2)c2c(nn1C)CCC2 N1(C(c2c(OC)csc2)=O)CCC(CNC(c2n[nH]cc2[N+](=O)[O-])=O)C(F)(F)C1 Cc1ccnc(CNC(C2CCC(CNC(=O)Cc3ccc(F)cc3)CC2)=O)n1 n1(CC(=O)NC2CC(NC(c3cnccc3Br)=O)C2)cc([N+](=O)[O-])cn1 C1(NC(c2c(COC)cccc2)=O)CCN(C(C2(C(N)=O)CCC2)=O)CC(C)(C)C1 C1(C(N2CC(C(C)C)C(C(=O)NCC(C)CC3CC3)C2)=O)CCCC(C#N)C1 C(=O)(CCC(C)C)NC1C(CNC(CC(=O)OCC)=O)C1 c1(C(N(C)CCNC(C2CCCOC2C2CC2)=O)=O)c(Cl)ccc2ncccc12 N1(C(c2cn(C)nc2C)C(=O)NCCCCCC)CCc2ccc(OCCC)cc21 CC(CCNC(c1cn(C)nc1C1CCCC1)=O)C(C)(C)C N1(C(c2c(F)ncc(OC)c2)=O)CCCC(C2(NC(C3(CO)CCC3)=O)CC2)C1 CCC(C)C(=O)C(=O)NCC#CC(=O)NCC1(C)CCCC1O c1(N2CC(CN(C(C(CC)=CC)=O)C)OCC2)nc(Cl)nc2c1ncn2C C1(C(=O)NCCOC2CCCC2)CC=CCN1C(=O)CCC1CCCOC1 N1(C(C(C)Sc2ccccn2)=O)CC2CC1CN2C(C12CC3CC1C2C3O)=O C1(NC(=O)CC2CC=CCC2)CCCCCC1NC(c1cc(CO)[nH]n1)=O CCC(CC)CCCC(=O)N1CCC(NC(=O)C(C)(F)F)CC2(CCC2)C1 C(=O)(C1=CC2CCCC12)N1C(C)C(NC(c2c(N)cc(F)cc2F)=O)CCC1 C1(CC(=O)NCCN(C(C)C)CC)CCCN1C(=O)CC1CNC(=O)C1 c1(C(N2CCCC(NC(c3c(N)cn(C)n3)=O)C2)=O)cccc2c1C(=O)NC2=O C1(C(=O)NCC(C2(O)CCN(C(C3CN(C)C3)=O)C2)C)CN2CCCN1CC2 C(C(C(C)C(C)C)NC(c1csc2nccn12)=O)NC(C)=O c1(C(N2CCC3(NC(C(CC)CC)=O)C(CC2)C3)=O)cnc2ccccc2c1 C(C(C)(C)C#CC(=O)NC1CC(O)C1(C)C)NC(c1cnc(OC)s1)=O CC1CN(C(=O)CCC2CCCCC2)CC1CCNC(C1CC=CCC1)=O C12CCCN(CC1)C(=O)COCCNC2=O.c1(OC)cnc(OC)nc1 C1(NC(Cc2nc(C)sc2C)=O)CC2(NC(C3CC3Br)=O)COC1C2 Cc1coc(C)c1C(=O)NCc1nc(C(=O)NOC2CCOC2)c(C)o1 C1(CNC(=O)Cc2ccc(Cl)s2)CC2(CCC2)CN1C(C1C2CCCOC12)=O c1(OCC)cc(C(N2CCOC(CNC(=O)Cc3csc(=N)[nH]3)C2)=O)ccc1C CN1CC2CC1CN2C(=O)CC1CCCN(C(=O)CCn2ccnn2)C1 c1(C(N2CCC(N(C(C)C=Cc3ccco3)C)C2)=O)cccc(Cl)c1Cl C1(C(=O)NCC(C2CC2)NC(CCC(=O)N(C)C)=O)CCCS(=O)(=O)N1 C1(NC(COC)=O)CC(CNC(=O)C(C)NC(=O)OCC2CCCO2)C12CCC2 C1(CNC(c2c(CC)cc[nH]2)=O)CN(C(=O)C(C)=C2CC2)CC(C(F)(F)F)O1 CCCCC(C(=O)N1CCC(C)(C(=O)NC2CN(C(C)C)C2)CC1)C(C)C N1(C(C2N(C(C3ON=C(CC)C3)=O)CCOC2)=O)CCOCC2(CC2)C1 c1(OC)ccc(CN2CC3(CC3)CC2C(=O)Nc2cccc(C)c2O)c(C#N)c1 N1(C(CCC2(C)N=N2)=O)CCC(NC(C2CCCCC2C(F)F)=O)C2(CCC2)C1 C1(CNC(C(Br)=C(C)C)=O)C(CNC(C2CC(C)(O)C2)=O)C1(F)F C1(C(N2CC(CC(C)NC(c3nn(C)c(Cl)c3Cl)=O)C2)=O)CC2CCCCN2C1 N1(C(C(C)(C)OCC)=O)CCC(NC(=O)CNC(C)=O)CC1 c1(SC)cccc(CC(=O)NCC23CC2CN(C(C2(F)CCOCC2)=O)C3)c1 c1(C(N2C(C(=O)NC(c3ncc(C)s3)CC)CC2)=O)ccnc(CO)c1 C(=O)(CC(C)(C)C(=O)N1CCCC(CNC(c2cc[nH]n2)=O)CC1)OCC c1(C(N2CCC(C)(NC(=O)Cc3cnccn3)CC2)=O)ccccc1C#CC1CC1 N1(C(CCN(C(C(CSC)O)=O)CC2CC2)=O)CCC(C)(C2CC2)C1 c1(OC)ncc(C(=O)NCC2CC(F)(F)CN2C(c2cc(C)sn2)=O)cc1C N1(C(C2C(C34CC(C(=O)NC(C)(C)C)(C3)C4)C2)=O)CC=C(CCCO)CC1 c1(NC(C(CN(C)C)O)=O)ccc(C(=O)NCC(F)(F)CC2CC2)cc1 C1(NC(CCC2CCN(C)CC2)=O)CCC2CN(C(C3COC(=O)N3)=O)CC2C1 c1(OCC)ccc(CNC(C2C(C(N3C(C(=O)OC)CCCC3)=O)C2)=O)cc1I C(CCOC)(C(=O)NC)NC(C1C(C(=O)OC)C1)=O.n1(CCCOCCO)ccnc1C c1(CC(=O)OC(C)(C)C)ccc(C(=O)NCc2cn(C3CC3COC)nn2)cc1 N1(C(c2cnn(C)n2)=O)CCC(C)(C)C(C(=O)NC2CC(OC3CC3)C2)C1 C12(NC(C=CSC)=O)CCCCCC1N(C(c1ccc3ccnn3c1)=O)CC2 C1(NC(c2c(CC)nc[nH]2)=O)C=CCN(C(=O)C(c2cccc(OC)c2)O)C1 Cn1cccc1C(=O)Nc1cccc(CNC(=O)C(c2cccc(F)c2)O)c1 CCC(COC)C(=O)NCCCCCCN(C)C(C1CCCCC1O)=O C(=O)(C1CCOc2c(F)cccc21)N1CCC(NC(C2(CSC)CC2)=O)C(O)C1 CC1CCN(C(C23CCC(C2)OC3)=O)CC1CNC(=O)CCc1ccn(C)n1 C(=O)(C1=COCC1)NCC1(CNC(CCc2cc(C(C)C)no2)=O)CCCC1 N1(C(CCc2cc(OC)no2)=O)CCCN(C(C2CC3CC4C(C3)C24)=O)C(C)C1 c1(C(=O)NCCN(C(C2C3CCCC23)=O)CC2CC2)coc2ccc(Br)cc12 c1(C(N2CC(C)C(NC(=O)CC3CCCOC3)C2)=O)ccc(S(N)(=O)=O)cc1F N1(C(C(C(CC)O)C)=O)CCCN(C(=O)CCCCCOC)CC1C N1(C(C2(NC(N)=O)CCC2)=O)CCCC1C(=O)NCc1nnc(CO)s1 c1(C(N2CC(CNC(C3CC4(CCC4O)C3)=O)C2)=O)cnc2c(F)cccn12 C1(NC(c2nn(CC)c(C)c2)=O)CC(C)CN(C(=O)C(C2CCOCC2)F)C1 N1(C(C2CCC(C)CC2)=O)CCC2(CCCCC2NC(c2sccc2F)=O)C1 c1(C(C(=O)NCCCCCC)N(C2CC2)CC)ccc(OC(C)(C)C)nc1 N1(C(CC(n2c(CC)ncc2)C)=O)CC(NC(=O)CC2(CSC)CC2)C(C)C1 c1(C(=O)NC2CC(CNC(c3c(C#C)cnn3C)=O)C2)scc2c1OCCO2 Cc1[nH]nc(C(=O)N(C(C)CCNC(=O)Cn2cnc(C(F)(F)F)n2)C)c1C N1(C(c2cc(C)cc(O)c2)=O)CCC2CCN(C(c3n[nH]c(C)c3O)=O)CC2C1 c1(NC(C2CCN(S(=O)(=O)C(F)F)CC2)=O)ccc(OC(F)(F)F)cc1C c1(CCCC(=O)NC2(CNC(C3CCC(CC)C3)=O)CCC2)cc(F)ccc1F N1(C(C2C(C)C2)=O)CCC2CN(C(c3ccc4cccnc4n3)=O)CC2C1 Cc1cc(O)ncc1C(=O)NCc1cc(C(=O)N(C)CCOCCO)n[nH]1 CC(C)CC(O)C(C)C(=O)NCCOC1CN(C(c2ncccc2C2CC2)=O)C1 Cc1ccn2c(=O)c(C(=O)NCC(C(C)C)NC(c3cnsc3C)=O)cnc2c1 c1(C(=O)NC2CC(N(C(c3c(OC)scc3)=O)C)C2)sc(C2CC2)nc1C N1(C(CCN(C)CCO)=O)CC(NC(c2ccc([N+](=O)[O-])s2)=O)CC(O)C1 N1(C(c2ccc3n[nH]cc3c2)=O)C2CCCC1CC(Nc1ncc(I)cn1)C2 N1(C(CCC(C)OCC)=O)CCN(C(=O)Cc2ccnn2CC)C(C2CCC2)C1 N1(C(c2c(OCC)cncc2)=O)CCOC(C)(CNC(C23CCCC2C3(F)F)=O)C1 N1(C(C2(C#C)CCC2)=O)CCCC(C2CCN(C(c3ncccn3)=O)C2)C1 c1(C(=O)NCCCCC(C)NC(CCC(=O)NCC)=O)ccc(=O)n(C(C)C)c1 C1(CNC(CCC)=O)CN(C(=O)Cn2nc(C(F)(F)F)cc2Cl)CCCO1 CC(CCCCNC(=O)CCCc1cnn[nH]1)NC(=O)CCC1CC1 C1(C(=O)Nc2cccc(NC(C3CCN(C)CC3)=O)c2)CC2CCCC2C1 c1(C(=O)NC2COCC2NC(C2CCC2(F)F)=O)nc2nc(C(F)(F)F)ccn2n1 N1(C(CCC=C)=O)CCN(C(C2CCn3cc(C)nc3C2)=O)C2CCC12 c1(OC)ccc(C(N2CCC(OC)CC2)C(=O)NC(C)C)cc1OC N1(C(c2c(C)n(CCO)cc2)=O)CC(NC(C23CCCC2C3)=O)CC(C)C1 Cc1cn2nc(C(=O)NC3(C)CCN(C(C4CCOC4C)=O)C3)cc2c(=O)[nH]1 CCC(N=c1nc(N(C)Cc2ccc(C)cc2Br)c2ncn(CC)c2[nH]1)C1CC1 C1(CC)C(=O)NCCN1C(=O)CCC1CCN(C(=O)CSC2CCOC2=O)CC1 c1(CC(=O)NCC2(CCNC(CCC(=C)C)=O)CC2)ccc2c(c1)CCCC2 N1(C(=O)CC2CCCC23CC3)CC(C2CN(C(c3cc(CO)[nH]n3)=O)C2)C1 C1(Nc2ncc(C(=O)OCC)s2)C(C)CCN(C(=O)CCCC2CCCC2)C1C C12(Nc3nccc(OCC)n3)CCCC1N(C(=O)CC1CCCC(OC)C1)CC2 CC(CN(C)C)CCC(=O)NC1(C)CN(C(=O)C2=NOCC2)C1 c1(N(C)Cc2nccn2-c2ccccc2)nccc(=NCCc2ccc[nH]2)[nH]1 c1(OC)c(CC(=O)NC2CC2CNC(=O)C(C)(C)CF)cccc1F c1(C(N(CCCC(=O)OC(C)(C)C)CC)=O)ccc2c(c1)c(C(F)(F)F)cn2C c1(C(N2CCC(F)(C(=O)NC(C)CN(C)C)CC2)=O)cc(N(C)C)cc(C#N)c1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC2C(NC(C3CCCN(CC)C3)=O)C(C2)C1 C(=O)(C1=CCCCC1C)NCC(CNC(COCCC)=O)(C)O N1(C(=O)OC(C)(C)C)CCC1CC(=O)NCC1CC(C(F)(F)F)C1 c1(C(=O)NC(C2CCCC2)CNC(CC(=O)NCC)=O)cscc1S(C)(=O)=O C(=O)(CCCC(C)C)NC1(C(N2CC(CC(=O)OCC)C2)=O)CC(F)C1 CCC(CC)CCCC(=O)NCCN(C(C1CC2C=CCC(C1)C2)=O)C(C)C C1(C(=O)NCC(CNC(c2c(C)nccn2)=O)F)CC2C(C1)C2(C)C c1(OC)cc(SC)c(NC(=O)CCC(F)F)cc1C Cc1ccccc1C(C)CC(=O)NCCNC(c1c(Cl)n[nH]c1C)=O CCC(C)CCCCC(=O)NCC(C)NC(C1(C(F)(F)F)CCCCO1)=O c1(C(=O)NC(C2CCCN2C(=O)CC2CC2)C)ccc(Br)cc1 c1(CC)ccccc1C(CNC(=O)C(C)CCOC)NC(=O)CC(C)(C)C c1(C(N2CCCC(CN(C(=O)CC3C=CCC3)C)C2)=O)ccc(=O)n(CCO)c1 N1(C(c2c(C)ccc(C)c2)=O)CC(NC(C2C3CCCC23)=O)CC12CCCCC2 c1(C(=O)NC2C(NC(C(C)O)=O)C2)ccc(NS(C)(=O)=O)c(Cl)c1 C1(CNC(c2cccc(C)n2)=O)CCCC2CN(C(c3cc(C)sn3)=O)CC12 N1(CCOC)CCCN(C(c2cnc(O)cc2C)C(=O)NCCCSC)CC1 N1(C(c2ncn(C)c2)=O)CC2(C(=O)NC3CCC4CC34)CC1CCO2 c1(NC(C2N(C(CCc3ccc(C)cc3)=O)C3C(C2)C3)=O)c(F)cc(Br)cc1F CN1CCCC1C1(N2CCCC2=O)CC1.C12CCCC1CCOC(=O)C2 N1(C(C(C)Oc2cccc(C)c2)=O)CCOC2CS(=O)(=O)CC12 C1(CC(=O)N(CC(CC)NC(c2scc(CC)c2)=O)C)CC2CCC1CC2 C(=O)(C1CSc2ccccc21)NC(C)CN(C1CCCC1)C(c1ncccc1N)=O CC(C)(C)C(=O)C(=O)N1CC2C(CNC(c3cccc(N4CC=CC4)c3)=O)C2C1 C1(C(N(C2CC(C(=O)NC3CCSC3)C2)C)=O)CCCC(CF)C1.CCO N1(C(C2(C)CCCN2C(=O)CC23CCCC2C3)=O)CCC2(CCCC2)C1 N1(C(c2cc(C)n(C)n2)=O)CC2CCN(C(=O)CC3CC3(Cl)Cl)CC(C2)C1 N12CCC(O)(C1)CC2=O.c1(-c2cn(C(C)(C)C(=O)O)nn2)cncc(Cl)c1 C12(NC(C3C(CNC(CCCNC(=O)OC)=O)CCC3)=O)CCC(CO)(CC1)C2 C(C(F)(C(=O)OCC1CC(=O)N(CCN(C)C)C1)C(C)C)NC(=O)OC(C)(C)C Cc1cc(Br)cnc1CNC(C1CC1C(=O)Nc1cccnc1)=O C1(C(=O)NCCC(n2cc(C3CC3C(=O)O)nn2)C)NC(=O)OC1C C1(NC(=O)C(c2ccccc2)=O)CN(C(C2CC3CC2C3)=O)CC12CC2 C1(NC(C2C=CCC2)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)c(F)c1)(F)F C(CCC(=O)N1CCCC1C(C)(C)C(=O)NC(C)C(C)CC)=CC O=C(C1=CS(=O)CCC1)NC1CC2(C1)CC(NC(C1CCn3ncnc3C1)=O)C2 C1(F)(CNC(C(CC)n2cccn2)=O)CCC(CNC(=O)C=CC2CCOC2)CC1 Cc1cn2c(=O)c(C(=O)NC(C)CNC(c3ccn4nccc4c3)=O)cnc2s1 CCC(CN(C)C)CC(=O)NCC1CCCCN(C(=O)C=Cc2cn[nH]c2)C1 Cc1nonc1C(N1CCC1CNC(c1occc1-c1ccccc1)=O)=O c1(C(=O)NC(C(C(C)C)C)CNC(=O)CSC(C)(C)C)ncnc2ccsc12 c1(CNC(C(C)OC)=O)cncc(C(N2CCC(n3ccnn3)C2)=O)c1 Cc1coc(C)c1C=CC(=O)NCC1CN(C(C2(C(N)=O)CC2)=O)CCO1 CN1CC(NC(C2CN(C(=O)C=Cc3ccsc3)CCO2)=O)C2(CC2)C1 c1(C(N(C)CCNC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)=O)cc2n(c1)CCCNC2=O C=CCCCCCCC(=O)NC(C)C(C)NC(=O)C(=O)NCCC(N)=O c1(C(c2nnnn2C(C)C)NCC(CSC)C)c(C)cnn1COC c1(-c2nc(Cc3ccc(Cl)cc3)on2)ccc2sccc2c1 N1(CC)CCN(c2ccc(NC(C3CC(C)C3(C)C)=O)cc2)CC1 C1(C(=O)NCC2(CNC(C(CC)C)=O)CCC2)CC2(CCCC2)C1 C(=O)(C(CC)(CC)OC)NCCC1CC(NC(C2CC(C#C)(O)C2)=O)C1 C12CCCN(C1CC)C(=O)C2.C#CCC(C(N)=O)n1cc(CCCCC(=O)O)nn1 N1(CCC)C(=O)CCC1C(=O)NCC(c1ccccc1)NC(c1cnn[nH]1)=O Cc1nc(C)n(CC(=O)N(C(c2ccccc2)CNC(C2(CCO)CC2)=O)C)n1 n1(CCOC)cccc(C(=O)NCC2CC(C)N(C(=O)C(C(C)C)SC)C2)c1=O C(=O)(CC(CC(C)C)N(C)C)N1C(C)(CC(=O)NC(c2nc(C)oc2C)C)CC1 C1(C(C)C)(CO)CCN(C(=O)C(C2CCCC2)NC(c2cc[nH]c(=N)n2)=O)C1 CCCC(C(=O)NCC1(CNC(C2(CO)CCCO2)=O)CC1(F)F)NC(N)=O C(C(=O)NCc1cccc(Br)n1)(C1=NOC2CC12)N(CCCF)C N1(C(C(C(C)C)C#N)=O)CCCC(C)(C)C1CNC(=O)CCOc1ccccn1 CC1CN(C(=O)CC(CNC(=O)C=Cc2cnccn2)C2CCC2)CCO1 C(CC(CNC(=O)Cc1cnc[nH]1)NC(=O)C(C)CSCc1ccccc1)OC CC1(C(N2CCC(CF)(NC(=O)COCC3CCOC3)C2)=O)CCNC1=O c1(C(N2CCN(C(c3cscc3C(F)(F)F)=O)CC2)=O)nccc2ccncc12 Cc1cc(C)c(CNC(C2CC(F)(F)C2)=O)c(C)c1Br N1(C(C#CC(C)C)=O)CCC(NC(=O)CSc2nccn2C)C2(CCC2)C1 N1(C(C2CC3(C(OC)CC3)C2)=O)C2CCC1CC(NC(=O)Cc1nonc1C)C2 Cc1ccc(-c2cn(CC3CC(CNC(C4CC4(C)C(F)F)=O)C3)nn2)nc1 N1(C(CN2CCC(C)(O)C2)=O)CCCC2(CCCN2C(=O)CC2CC2(C)C)C1 c1(C(=O)NCC2CCN2C(C2CC(O)(C(F)(F)F)C2)=O)cc(=O)n2ccsc2n1 CC1CCC(CNC(C2NC(=O)OC2C)=O)CN1C(=O)C=CC1CC1 n1(CC(=O)NC2CCC2CNC(c2cccc(C3CC3)c2)=O)ccc(O)nc1=O C1(C(=O)NC)CC(O)CN1C(=O)C(C1CCCN(C(=O)CCCCN(C)C)C1)C CC1CC(Cc2ccccc2)CCN1C(c1nc(C(F)F)ccc1Cl)=O C1(CC=C)(C(=O)N(C)CC2CCCC3CC23)CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 C1(Cc2ncc(C(=O)OC)nc2)CCC(C(=O)Nc2c(CSCC)ncs2)CC1 CC1(C)CC(NC(=O)C2=CCCCC2)CN1C(=O)Cc1ccc(Cl)c(F)c1 CC1(C)CC(CC(N2CCOC(CNCC3CC34CC4)C2)=O)CO1 C1(C(=O)OCC)CC(CNC(C2CCC(NC(C)=O)CC2)=O)=NO1 O=C1CCC(CCC(N2CC(O)(CNC(=O)CC3CSC3)C2)=O)N1 Cc1cc(C)c(CC(C(=O)O)NC(C2Cc3cscc3C2)=O)c(C)c1 c1(CC)cc(C(N2CCC(F)(CNC(C3CC(CC(C)C)C3)=O)C2)=O)c(C)nn1 N1(C(c2c(C)nc[nH]2)=O)CCC(NC(C2CCCN(C(C)C)C2)=O)CC(C)(C)C1 CCC(C)CC(C)C(=O)NC1(CC=CC(=O)NC2CC3CC2CC32CC2)CCC1 N1(C(C=CC(=O)OC)=O)CC23CCCC2(C1)CN(C(c1c(C)coc1C)=O)C3 c1(C(=O)NCC2C(CNC(c3c(C#C)c[nH]n3)=O)C2)ccc2c(=N)[nH]cnc2c1 N1(C(c2cc(C)cc(O)n2)=O)CC(NC(=O)CCCC#N)CC12CCCCCC2 Cc1ccc2oc(C(N3CC(NC(=O)CC4CCCCC4O)C(C)C3)=O)cc2c1 CCC(C)(CCNC(=O)C(C)C(F)F)NC(C1SCC=C1C)=O C=CCCCC(C(=O)OC)NC(=O)CCOCCCNC(=O)C(F)C(C)(C)O c1(C)cn(C)c(C)n1.C1(O)(C(C(=O)NCC2(CC)CCC2)F)CN(C(=O)C2CC2)C1 C1(SC)CN(C(=O)C(F)(F)c2cn[nH]c2)CC1NC(=O)C(C)C C(=O)(CC(F)(F)c1ccncc1Br)NCC(C)CN1CCCC1=O Cc1ccc(C(N2CCCCCC2C(=O)NCC(C)(C)C2CC2)=O)c(F)c1 c1(C(N)=O)cnccc1Br.c12cn(nn1)C1CCN(C1)CC(=O)NC2.C1(=O)CN1 C1(CC(=O)NC(CNC(C(CCOC)C)=O)(C)C)CSc2ccccc2O1 C1(O)(CC#C)CCN(C(=O)CCNC(CC(C)(C)n2ccnc2)=O)CC1 c1(NCC(=O)NC2CCN(Cc3ccn(CC)n3)C2)ccc(Cl)cc1Cl N1(C(C(c2cccnc2)C)=O)CC2CCC(C1)N2C(c1cnc(O)n(C)c1=O)=O C1(C(N2CC(C(N(CC)Cc3ccoc3)=O)C(F)C2)=O)CCC(C)(C)CC1 N1(Cc2ccsc2)CCCS1(=O)=O.n12cc(nn1)C(C1CC1)NC(=O)C2 Cc1c(C(N2CCC(c3cn(CCO)nn3)C23CCC3)=O)sc2ccc(Cl)cc12 c1(CNC2CCC(C(=O)NC(C)CN3CCCC3)C2)cc(Cl)cc(Cl)c1 Cn1cc(NC(C2CCCN2C2(COC(C)(C)CO)CN(C(=O)C3CC3)C2)=O)cn1 N1(C(C2CC(C(C)(C)C)C2)=O)CCCCC(CC(=O)NCC2C3CCCOC23)C1 Cc1ccc(OCC(=O)NC2CN(C(c3cc[n+]([O-])cc3)=O)CC2(C)C)cc1C Cn1cnc2sc(C(=O)NC3(C)CC(NC(C4CCS4(=O)=O)=O)C3)cc12 C(=O)(CCCCCn1cc(CO)nn1)NC1(C(N2CC(CC)OCC2)=O)CCSC1 N1(C(C2(CC)CCN(C(=O)C=C=C(C)C)CC2)=O)CC(OC)CC(F)(F)C1 C1(CNC(c2c(C)ocn2)=O)CC(C)(C)CN1C(C12CCCCC1C2)=O C1(C(N(C2CN(C(=O)C(C)(O)C(F)(F)F)CC2(C)C)C)=O)CCC2(CCC2)CC1 C1(O)(CCNC(c2c(CC)[nH]cc2)=O)CCCN(C(=O)C(CC)n2ccnc2)C1 Cc1cc(C(N2CCOC(C3(C)CC3)C2)C(=O)NC2CC2)cc(C)c1 c1(N)ccc(F)c(C2(C)CC2)c1.c1(C(=O)NCC2C(C(=O)OC)C2)cc(Cl)ccn1 C(=O)(CC(C)(C)C(F)(F)F)NCC(CNC(C12C(C)(C)OCC1C2)=O)O C1(Cc2cn(NC(CC3CCC(C)C3)=O)nn2)CCC(CO)CC1 c1(C2CCN(C(c3cccc(CC)c3)=O)C2)ccc(OC)c(OC(F)F)c1 c1(CN(C(c2nonc2C)C(=O)NC(CC)(C)C)C)nnn(C)c1C CC(C)CC(O)C(C)C(=O)N(CC(C)(C)NC(C1(c2cc[nH]n2)CCC1)=O)C c1(CC(=O)NC2CN(C(=O)C(c3cccc(F)c3)F)CC2F)cccc(F)c1Cl C(=O)(CCCCCN=[N+]=[N-])N1C(C(=O)NC(C=C)(C)C)CN(C)CC1 N1(C(C(C)(C2CCC2)NC(CSCC=C)=O)=O)CCC2(CNC(=O)N2)C1 Cc1cc(C(N2CC3(CNC(=O)C4=CCCC4C)CCC2C3)=O)c(O)nn1 C1(C(=O)NCC2(CCNC(C3C(C(=O)OCC)C3)=O)CC2)COC2(CCC2)C1 N1(C(Cc2nnc(C)o2)=O)CC2CC1C2NC(c1ccsc1Cl)=O c1(C(N2CCC(C)(C)C2NC(=O)CCCC(F)(F)F)=O)ccc2ccncc2c1 C(=O)(C1=CC2(CCN(C(=O)CC3CCC3)C2)C1)NCC(CC(=O)OC)O c1(CCC)ccc(-c2csc(C(=O)Nc3cc(O)nc(Cl)n3)n2)cc1F N1(C(c2cc(OCC)n[nH]2)=O)CCCCC(N(C)C(C2CC2(C)C(F)F)=O)C1 Cc1cccc(C(O)C(=O)N(CCCNC(c2ccc(Cl)s2)=O)C2CC2)c1 C=C=C(C)CC(=O)NC1(C2CCCCN2C(=O)CCc2ccc[nH]2)CC1 c1(C(N2CC(C)C(N(C(=O)C3=CCC3)C)CC2)=O)ccn2c1CSCC2 Cc1oc(Br)cc1C(=O)NC(CNC(c1c[nH]c(C(F)(F)F)c1)=O)CO c1(C(N2CCC(CCNC(C3NC(=O)OC3)=O)C2)=O)cccc2c1COCCN2 c1(C(=O)NCC2(CC(=O)NC3CN(C)C4C3C4)CC2)cn(C)c(=O)n1C N#Cc1ccc(NNC(=O)OOCOc2cccc(F)c2)cc1F c1(N(CCC(C)OC)C)nc(SC)c(C)c(=NC2CCCOc3cc(Br)ccc32)[nH]1 c1(CC(=O)N(CC(CC)NC(=O)C(COC)OC)C)ccccc1Br Cc1sc2ncnc(C3CCCO3)c2c1C.C(=O)(CC(C)C(F)F)N1C(CO)C1 N1(C(CCOC(C)C)=O)CCN(C(c2ccc(C(C)(F)F)nc2)=O)C(C(F)F)C1 Nc1cc2c(cc1C(N1CCC(CC(C)NC(C3CC3F)=O)CC1)=O)OCCO2 C1(CC)(NC(c2ccc(C3CC3(F)F)cc2)=O)CCN(C(=O)CC2CSC2)CC1 Cc1ccc(COC2CCCC3(CC2)CC3)c(F)c1F.c12nnnn1NC2C1CC1 c1(C(N2CCC(O)(CNC(=O)CC3CC34CC4)C2)=O)cc2cc(Cl)ccc2[nH]1 CCCC(C(=O)N(C)CC1CCCN1C(=O)C(CC)c1ccccc1)OC C1(NC(CC(C)OC)=O)CCC2CN(CCC3CC3(Cl)Cl)CC2C1 C1(C(=O)NC2CC(NC(=O)CCC3CCCO3)C2)(OC)CCOC1 CC1CN(C(=O)Cn2cccnc2=O)CC1CNC(=O)Cc1nc[nH]n1 c1(SCC(=O)NCCN(C2CC2)C(c2cc(C3CCC3)no2)=O)cccc(O)c1 Cc1cc(NC(C2(C)CCCS2)=O)ccc1NC(c1nc(C)ncc1Cl)=O C=Cc1cncc(C(N2CC(C)(C(N3CCCCCC3)=O)C2)=O)c1 C(CN=c1nc(N2CCC3(CCOC3)C2)c2sccc2[nH]1)N1CCC(CO)C1 C1(OC)(CNC(=O)C(C)S(N)(=O)=O)CCN(C(=O)Cc2ccnc(C)c2)CC1 C(=O)(CCC(CC)OC)NC(C(=O)NC(CCC)CC)CC1CCC1 C(CCC)(CC(=O)OC)NC(N(c1ccccc1Br)CCCC)=O Nc1ncccc1C(N1CCCC(NC(C2CNC(=O)N2)=O)C1)=O C(CCCCC(=O)N(C)CC1OCCC1(C)C)NC(C1(CCC=C)CC1)=O N1(C(CCSCCCC)=O)CCC(NC(=O)COCc2ccnc(O)c2)C1C C1(C(N2CCCC(C(C)NC(c3c(C)scc3)=O)C2)=O)CC(C)(C)OC(C)(C)C1 c1(C(=O)NCC2(F)CC(NC(C=C(C)Cl)=O)C2)ccc2c(c1)NC(=O)CN2C C1(CC(=O)NCCCCNC(C2(C)C(C)(C)C2)=O)COCC1(C)C c1(C(N2C(CNC(c3c(CC)occ3)=O)COCC2)=O)cc(F)c(N)cc1OC c1(C(N2CC(C(=O)Nc3c(C#N)cc(CC)s3)C2)=O)ccc([N+](=O)[O-])c(C)c1 c1(OC)ccc(C(=O)NCC2C(C)CCCN2C(c2csnc2Cl)=O)c(F)c1 c1(OC)nc(C(=O)NC(C)CC(C)NC(=O)C=Cc2ncc[nH]2)ncc1F c1(NC(=O)CN2CC3CCCC3C2)cccc(S(=O)(=O)NC2CCS(=O)(=O)C2)c1 c1(C(=O)NC2(C)CCN(C(C3(c4ccccc4)CC3)=O)C2)[nH]nc2ncccc12 C(=O)(C1=CCCC(C)(C)C1)NCC(C)CNC(c1cc(CO)n(C)n1)=O C1(C(N(CCC(C)NC(COCCCC#C)=O)C)=O)=CC=CC=CN=C1CC C1(C(=O)NCC(N(OC)C)=O)(NC(=O)CCOC(C)=O)CCC(C)(C)C1 c1(C(N2CCC(CNC(C)=O)C(C)C2)=O)cc2oc(C)cc2[nH]1 CC(C)CC(C)(CNC1CC(OC(C)(C)C)C1)Nc1cc(-c2cccs2)ncn1 c1(C(=O)NCC2N(C(C(C)SCCCC)=O)CCC2)cnc(O)c(C(F)(F)F)c1 C1(NC(C(C)Cc2ccccc2)=O)CC(C)N(C(c2nccn2C)=O)C1 C(=O)(C1CCCc2ccccc21)NCC1CC(NC(c2csc(Cl)n2)=O)C1 c1(C(N2CC3CN(C(COCC)=O)CC(C2)O3)=O)coc2ccc(OC)cc12 c1(CC)cc(C(=O)NCC2CCCCN(C(C3CCN(C)C3)=O)C2)ccc1Cl C1(C(=O)NCCNC(=O)NC(C)C)CCOCC1C.C12CCC(C1)CN2 C(CCCCC(=O)N1CC(C)CC1C)c1ccc(OC)cc1 CC(C)C(CC(=O)NC(C)C(C)F)NC(c1coc(CO)c1)=O c1(C(N2CCCC(C(=O)NCCOC)C2)C(=O)NC(CC)C)sc(=O)n(C)c1Cl N1(C(CNC(C(CC)C)=O)=O)CC2CCC(N(C)C(C3CCN3CC)=O)C2C1 C12(C(=O)NCCN(C(C3(c4cccs4)C(C)C3)=O)C3CC3)CCCN(CC1)C2 C1(CN(C(C(Cc2cc[nH]n2)NC(C(C)OCCOC)=O)=O)C)CCCCCC1 c1(N2CC(CNC(C(CCCC)C)=O)OCC2)cc(SC)ccc1[N+](=O)[O-] c1(OC)cc(CC(=O)NC(C)Cn2cc(C3(O)CCCCC3)nn2)ccc1C Cn1ccc2c(-c3nc(C(F)F)nn3CCC3CCCCC3)ccnc12 c1(C(c2n(C(CC)C)nnn2)NC2CC(CO)C2)c(Cl)cccc1Br c1(C(C(=O)NC(c2cn(CC)nn2)CCC)C2CC2)cccc(I)c1 N1(C(c2ccn(CCF)n2)=O)CCN(C(=O)C(=CC2CCCCC2)F)C(CF)C1 CC1CCN(C(C2(C3(C)CC3)CC2)=O)C(C(=O)NCC2CN3CCC2CC3)C1 c1(CCC(C)C)ccc(C#CC(=O)Oc2ccc(Cl)cc2)cc1 Cc1cc(NC(=O)CC2CCN(C(c3cccc(F)c3)=O)C2)cc(Br)c1 CC(C)(CO)C(=O)NCc1cccc(NC(=O)CC2OCCO2)c1 CC1(CC(=O)NC2CC(NC(=O)CC3CCCOC3)C2)CCCCC1 CC1CCN(C(=O)CCOC2CCC2)CCN1C(c1coc(-c2cccs2)c1)=O n1(CCC(=O)NCCNC(C2(CC(C)C)CCOC2)=O)c(-c2ccsc2)nnc1S Cc1nc2c([nH]1)C(C(=O)N1CCCCC1CNC(=O)CN(C)C(C)C)CCC2 CCCC(C(=O)N(C)CC1(O)CN(C(C2(C)CCCOC2)=O)C1)NC(C)=O C(N=c1[nH]c2ccc(O)cc2s1)C(N1CC2c3cnc(nc3)C2C1)=O.C1CC1 N1(C(c2ccc(-c3nc(=N)s[nH]3)cc2)=O)CCCC2(COCCN2)C1 C1(N(C)C)CCC(C(=O)NCCNC(=O)CCc2cnoc2)C1 c1(C(=O)OC)ccnc(C(=O)N(C2C3CN(C(C4CC(C)(C)O4)=O)CC23)C)c1 N1(C(CC(CC)C)=O)CCN(C(=O)COCCF)CC1CF c1(C(=O)NCCCC2CCCCN2C(c2ccc(Cl)cn2)=O)csc2nnsc12 CCCC(=O)C(=O)N1CCCC(C2CCCN2C(c2oc(C)nc2C)=O)C1 c1(NC)nc(C)ccc1C(N1CC(CNC(=O)CCC2CCOC2)C(C)C1)=O C1(O)(CN(C(C2(CC=C)CCC2)=O)C)CCN(C(c2cncc(C)n2)=O)C1 C1(CNC(C2CCC(=O)N2)=O)CN(C(c2ccc(-c3cnco3)cc2)=O)C2CC12 Cc1ccc2c(C(=O)NCC(C)CNC(=O)CN(c3ccnc(Cl)n3)C)onc2c1 Cc1noc(C)c1CCNC(C1(NC(=O)CCc2nncn2C)CC1C)=O CC(CN=c1ccc(Br)c(S(=O)(=O)NC2CC2(C)C(F)F)[nH]1)C(F)(F)C(F)F C1(N(C(c2c[nH]nc2C2CC2)=O)CC)CCCN(C(=O)CC2(C)CC2)C1 C1(CCC(=O)NC(c2cn(C)nc2)C(=O)NCc2ccon2)CC(C)(C)CO1 C(=O)(C(F)(F)C(F)F)N1CC(CN(C(=O)COCC2CCOCC2)C)OCC1 Cc1cccc(C(N2CCC(CNC(C3CCC(C)(C)OC3)=O)C2)=O)c1[N+](=O)[O-] C=CC(CCC)CC(=O)NC(c1ccccc1)CNC(c1ccc(O)cc1)=O c1(C(=O)NC2CC(CCNC(Cc3ncc(C)[nH]3)=O)C2)cc(Cl)ncc1N c1(C(=O)NCC(c2ccccc2)N(C(CC(C)O)=O)C)cc(N)c(F)cc1F N(C1CCCn2ccnc21)C(C1(C)CCN(C(c2cccc(SC)c2)=O)C1)=O C1(C(N(C2CCN(C(CCC(=O)OCC)=O)CC2)C)=O)CCCC2CCCN12 C1(C(N(C)CC2N(C(C(CCCC)O)=O)CCC2)=O)CCN2CCOCC12 c1(NCC(=C)CC)nc[nH]c(=NCc2ccccc2SC)c1C CCCCCC(O)CC(=O)N1CC2(C1)SCCC2NC(C1CSCCS1)=O N1(C(C2C=C(C)CS2)=O)CC2(C(N3CCC4(CSC4)C3)=O)CC1CCO2 c1(OC)ccc(C(N2CCC(n3cc(Oc4ccc(Br)nc4)cn3)CC2)=O)cc1 c1(CC)ccc(C(=O)NCCC2CC(NC(c3occc3C)=O)C2)c(C)n1 c1(C(N2CCCC(N(C(c3n(CC)ccn3)=O)C)C2)=O)ccc(O)cc1C c1(C(N2C(CNC(CC3CC(C)(C)OC3)=O)CC2)=O)cccc2c1CC2=O c1(OC)cc(C(=O)NC2CC(CO)N(C(c3cc(O)n(C)n3)=O)C2)c(Cl)cn1 c1(C(=O)NCCCN(C(=O)CCCCN(C)C)CC)ccccc1[N+](=O)[O-] c1(C(N2CC(n3cc(C(CC)O)nn3)C(C)C2)=O)c(F)ccc2c1OCO2 c1(C(N(C2CCN(C(c3ccc(C4CCC4)nc3)=O)C2)C)=O)cccc(=O)o1 N1(C(c2ccc(C#C)cn2)=O)CC2(CCCC2NC(C2(CC)CC2)=O)C1 c1(OC)ccc(C(=O)NCCC(C)CCNC(=O)CSc2cccs2)nc1OC C1(CNC(CC(CC)SC)=O)CC2CCC1N2C(C12CC(F)(C1)C2)=O N1(C(CC=CCC)=O)CCC(C)C1CNC(C1(Br)CC1)=O.C1(C)(N)CCCC1 C1(C(=O)NCCCNC(C(COC)(C)O)=O)CCOCC12CCCC2 C1(C(=O)NCc2cc(C(C)C)ncc2)CCC2CN(C(=O)OCC)CC2O1.C(C)(C)(C)O C(=O)(CCS(C)(=O)=O)N1CCC(N(C(c2c[nH]c(C(N)=O)c2)=O)CC)CC1 c1(C(N2CCC(C)(CNC(CC=CC=C)=O)C2)=O)ccc2c(c1O)CCC2 c1(OCC)cc(NCc2ccccc2C(C)(C)C)ccc1OCC N1(C(c2cccc(C)c2N)=O)CCN(C(=O)CC2CCCN(C)C2)CC(CO)C1 Cc1cc(C)c(C(N2CC3(NC(C4CC5CC5C4)=O)CCC2CC3)=O)c(C)n1 Cc1ncn(C)c1C(=O)NC1CC(C)(CNC(=O)CCc2cncnc2)C1 C1(CNC(CCC=C=C)=O)(OC)CCN(C(c2ccccc2C(F)F)=O)CC1 CN=c1ccc(C(N2CCC(O)(CCNC(=O)CC(C)N(C)C3CC3)C2)=O)c[nH]1 C1(NC(CC)=O)CCN(C(C2(C(N3CCCC3)=O)CCCCC2)=O)CC12CCC2 C1(CNC(CC(C)n2cccn2)=O)CCC12CCN(C(C1(O)CC1)=O)CC2 c1(CC)ncc(C(=O)NCCCC(C)NC(=O)C(F)(F)c2cnn(C)c2)o1 N1(C(C(=O)NC)=O)CC23CCCC2(C1)CN(C(=O)CCC#Cc1ccccc1)C3 C1(CO)CCC2(CCN(c3nnnn3CCOc3cccc(Cl)c3Cl)C2)C1 Cc1ncc(C)c(NC(C(C)NC(=O)C(F)OC(F)(F)F)C(C)C)n1 C(=O)(C(CO)C(C)(C)C)NC(C1CCN(C(c2nc(CC)sc2)=O)CC1)C c1(C(=O)NC2CCC(CNC(Cc3c(C)occ3)=O)C2)cc(O)ccc1F c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CCC2)cnn2c(=O)cc[nH]c12 C(C1OCc2ccccc21)NC(=NCC=C)NCC(c1ccncc1)O C(C(=O)NCCCN(CCCNC(=O)CC1CCSC1)C)(C(C)(C)C)NC(C)=O CC(CCNC(C1C(C)C1C)=O)N(C(=O)Cc1nnnn1CC1CCOCC1)C C12(C)CC1C(=O)NC1CC(C1)CCNC2=O.C1(CC)(CN(C)C)CCC1 CC(CC(F)F)C(=O)N1C2CCC(C2)C1CNC(c1cnn(CC2CC2)c1)=O C12(CNC(CCCNC=O)=O)CCCCC1CN(C(=O)CCOC1CCCC1)C2 N1(C(=O)CN2CC=CC2)CCCC1C1CCCN1C(C1CC2(CCCC2)CO1)=O c1(C(=O)NC(CN(C(=O)CC(C)c2ccccc2)CC)C)cnc(S)[nH]1 c1(NC(C)C(c2ccncc2)O)ncc(S(=O)(=O)N2C3CCC2CSC3)cc1Cl C(C(CC(=O)N(C1COC(C)(C)C1)C)NC(c1cc(Cl)cs1)=O)OC c1(C(=O)NCCN(C(=O)C=CC2CCOCC2)CC)ccnnc1C C1(C(=O)NCCC=C=C)CC(C)CN(C(C2(SC)CC2)=O)C1 N1(C(C(CCSC)O)=O)Cc2ccnn2CC(NC(=O)Cc2ccccc2C)C1 c1(CCC(N2CCC(O)(c3cn(CC(=O)OC)nn3)C2)=O)cc(F)ccc1Br CC1CC(C(=O)NCCN(C(=O)CC2CCC(C)(C)O2)CC2CC2)CCO1 CCC(C)CCCC(=O)NCC1CC(O)CN1C(c1nccc(Cl)c1F)=O N1(C(CCN(C(=O)CSC(F)F)CC#C)=O)CCC(C(C)(C)O)CC1 c1(OC)cc(F)ccc1C(N1CC(NC(C2CCNC(=O)C2)=O)CC(C)C1)=O c1(C(=O)NCC(CO)NC(C2(COC)CC2)=O)csc2cc(Cl)ccc12 Cc1cccnc1C(N1CC(NC(c2ccc(-c3cc[nH]n3)s2)=O)C2CC12)=O C1(NC(C(C)(C)CF)=O)CC2CN(C(=O)Cc3ccoc3)CCN2C1=O N1(C(C(c2c(OC)ccc(Br)c2)(F)F)=O)CCn2c(CC(C)(C)C)nnc2C1 C12(C(N(CCCN(C(c3ccnc(OC)n3)=O)C)C)=O)CCCCC1C2 C=CCCCCC(=O)N1CC(CNC(=O)C(C)(C)c2csc(C)c2)C2(CC2)C1 C12(CNC(C3(NC(N)=O)CC3)=O)CCCC1CCN2C(c1cnc(C(F)F)s1)=O N1(C(C(c2cccc(N)c2)(C)C)=O)CCC2(CCCN2C(C2C=CCC2)=O)CC1 N1(C(C)C)CCN(C2CCN(C(C3CCCCN3CC3CNC(C)C3)=O)C2)CC1 N1(C(=O)NCc2c(CC)c(F)ccc2)CCN(S(=O)(=O)NC(C)(C)C)CC1 N1(C(c2cncc(N(C)C)c2)=O)CCC2C(C1)CN2C(=O)C(F)=C1CCCC1 N1(C(c2nc(-c3ccn(C)n3)sc2)=O)CCN2CCN(C(=O)CC3CC3)CC2C1 C12(NC(CN(C(=O)OCC=C)C(C3CCC3)C3CC3)=O)CCCC1OCC2 C(=O)(C1CCc2cccnc21)NC1C(NC(=O)CCn2ccc3cccnc23)C1 C1(CNC(c2n(CC)ccc2)=O)CCC2CN(C(=O)CCc3nc(=O)o[nH]3)CC12 c1(C(=O)NCCOCCNC(=O)CCCc2cccs2)ccc(C2CC2)c(F)c1 C1(OC)CCC(C)N(C(=O)CC=CCNC(=O)CCn2cccc2)C1 c1(CNC(c2c(CC)c[nH]n2)=O)nc2c(s1)CN(C(c1sccc1CC)=O)CC2 N1(C(c2cccc(C)c2)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCCC1=O)C3 N1(C(c2c(CC)con2)=O)CC(NC(c2coc(C)c2)=O)C(C)C1 N1(C(CSCCN(C)C)=O)CC(NC(c2cc3c(s2)CCC3)=O)CC(O)C1 c1(C(N2CC(F)(CNC(C(C(C)C)NS(C)(=O)=O)=O)C2)=O)nc(C)c(C)nc1C c1(NC)cc(C(=O)NCC(O)CNC(c2c(C)cccc2C)=O)cc(Cl)n1 CN1C(=O)c2ccccc2C1C(=O)NCC1CC(NC(c2cc(=O)cc[nH]2)=O)C1 CC1(C)CCCC(C(=O)NCC2COCCN(C(C3(C(F)F)CCCO3)=O)C2)C1 C1(C(C)NC(C)=O)CCCN(C(=O)C2CC2)C1.C(CON)SCSC c1(C(=O)NC2CC(C)(NC(CSc3nnc(C)s3)=O)C2)ccc2c(c1)NCC2 N1(C(c2c(C)nn(CCO)c2)=O)CC(NC(=O)Cc2c(Cl)cnn2C)CC(C)C1 c1(N2C(C(N3CCC(C4CCCN4C(=O)C4CC4)C3)=O)CCC2)ncc(F)cn1 CC(C)CC(C)(C(=O)NCC1CC(C(C)(C)C)=NO1)NC(=O)OC(C)(C)C C(C(=O)N=c1cc[nH]cc1)n1c(C(N2CCC23CC(n2ccnn2)C3)=O)ncc1 Oc1ccc(CNCC2CCCN2Cc2cc(Cl)ncc2Br)c(F)c1 N1(CC=C)C(=O)NC2C3=C1CC1CCC31CCC(=O)N1C=CC=CC=C1C2CC C#Cc1ccc(C(=O)NCC2CCCCC2C(=O)NC23CCC(C2)OC3C)cc1 N1(C(Cc2c(OC)ccnc2)=O)CCC(NC(=O)CN=S(C)(C)=O)C(C)(C)C1 CC1CN(C(=O)C(=O)Nc2ccon2)CC1CCNC(=O)C(N1CCSCC1)C C(=O)(C1=C(C#N)CCC1)NCC(=O)NCC(=O)NCC1(CC)CC(C)(C)C1 N1(S(CC2CCC(C)O2)(=O)=O)CCc2c(ncn2C2CCCC2)C1 Cc1ccc2c(C(N3CCCC4(C3)CN(C(C3COC(=O)O3)=O)C4)=O)c[nH]c2c1 CC(CC(=O)N1CCC(F)(CO)CC1)C(C)(C)NC(=O)C(F)OC(F)(F)F C1(NC(c2c(Cl)ccc(C)c2)=O)CC2CC(C1)N(C(C1CCCN1C=O)=O)C2 CC1=NS(=O)(=O)N(CCC(=O)N(CCNC(=O)COCC(C)C)C(C)C)C1 C1(C(N(CC(C2CCCC2)O)C)=O)(NC(=O)CC2CCCC3CC23)CC(F)(F)C1 Cc1cc(C(=O)NCC(C)(C2CCC2)NC(=O)C(C)SC(F)(F)F)c(C)o1 c1(C(N2C(C)CC(CNC(c3c(C)nn[nH]3)=O)C2)=O)cccc(=O)n1O CCC(CC)C(F)C(=O)N1CCC(O)(CCNC(c2cccc(CO)c2)=O)C1 CC(C)(C)CC(O)C(=O)NC1CC1NC(=O)Cc1csc(=N)[nH]1 c1(C2(C(=O)NC3CCN(C(Cc4ccc(C)s4)=O)C3)CCC2)cnccc1C N1(C(=O)COc2ccc(CN3CCOC3=O)cc2)CCC(F)(F)C(O)C1 n1(CCNC(C2(F)CN(C(C3C(C)(CC)C3)=O)C2)=O)nc(C)nc1C C(C(C)(F)C(C)(C)F)(c1nnnn1CCC)NCc1ccc(OCCCC)cc1 N1(C(c2scc(C)c2Br)=O)CCN(C(=O)CCCCC(C)C)CCC1C c1(OCC)ccc(C(=O)NCC2CC2NC(=O)CC2OCCC2(C)C)cc1C.OCC C(=O)(CC1CCc2ccccc21)NC(C)CNC(c1cnc2c(c1)NC(=O)CO2)=O c1(OCCN(C(=O)C(O)C(O)c2ccccc2)CC)ccc(CC#N)cc1 O=S(=O)(c1ccc(NCCF)cc1Br)NCC1CCN(Cc2ccccc2)C1 c1(CC)csc(C(=O)NCc2ccc(C(=O)NCC3CC3C)o2)c1 c1(C(=O)NCC(C2(CC)CCCC2)=O)cc2c(nn1)CCOC2 c1(NCCCCCN(C)C)ncccc1S(=O)(=O)NC1CCC12CCC2 c1(C(=O)NCc2c(SC)cn(C)n2)c(C)ccc(Cl)c1O C=CCC(CC(=O)NCCn1cnnc1C)NC(C1(C#N)CCCOC1)=O C(CNC(=O)C=Cc1cccc(OC)c1)(CC(F)(F)F)NC(C(C=CC)O)=O Cn1ccc2cccc(CN3CCC(C(=O)NCCc4cc[nH]n4)C(O)C3)c12 N1(C(c2ccc(C)cn2)=O)CCC(C(=O)NC2C3COCC23)C12CC2 c1(OCCC)cccc(CC(=O)NC23CC(NC(c4cc(=O)cc[nH]4)=O)(C2)C3)c1 C1(NC(c2c(C#N)cn[nH]2)=O)CC2(NC(=O)Cc3ccc(Cl)cn3)COC1C2 N1(C(CC2(C(=O)OC)CC2)=O)CCC(O)(C(C)NC(=O)CCCN(C)C(C)=O)C1 N1(C(CC=CCCCCC)C(=O)NCC2CCOC2)CCC(C)(F)CC1 C1(CNC(C(C)OCCOCC)=O)CC2CCC1N(C(C1(C)C=CCC1)=O)C2 CC1CN(C(=O)C(N2CCCC2C2(C)CC2)=O)CCN1C(=O)CC1CCCCC1 C1(C(N2CC(CNC(=O)C3=CCCC3)C(O)C2)=O)CCCCC1(F)F c1(OC)ccnc(Cl)c1COC(SC(F)(F)F)=O c1(C(N2C(CC(=O)NC(C(C)SC)C)CC(O)C2)=O)cc(C)c(C)nn1 C1(NC(C2(OC)CCC(C)C2)=O)CC2CCC1CN2C(C1C2CC3C(C2)C13)=O CC1CC(NC(=O)CCN2CCCC2)CCN1C(C1CCCC(F)(F)C1)=O CCC(C)CC(=O)C(=O)N1CC(C(=O)NC2(COC)CCC2)C(C)C1 N1(C(C(c2ccc(C)cc2)C2CC2)=O)CCC2CCC(C1)N2C(=O)CN(C)C C1(CNC(C(C2CC2)SC)=O)(NC(c2cc(C#N)c[nH]2)=O)CCCCC1 C1(NC(C2CC23CCOCC3)=O)CC12CCN(C(c1cc[nH]n1)=O)CC2 C1(C(=O)NC2CCC2O)CC12CCN(C(=O)Cn1cc(CO)nn1)CC2 C12(NC(c3cn4c(n3)SCC4)=O)CCOCC1CN(C(C1CCCCO1)=O)C2 n1(SCC(CC#N)O)ccc2cc(C(=O)O)ccc12 C#Cc1c[nH]nc1C(=O)NCC(C)N(C)C(c1cnoc1C1CC1)=O C1(C(=O)NCCNC(=O)OCC)CCCCN1C(=O)Cc1nc(C#N)cs1 c1(C(=O)NC2(C)CC(NC(C34COCC(C3)C4)=O)C2)nc2ccccn2c1F C1(C(=O)NCC2(N3CCCC3)CC2)CCCCC1NC(c1c[nH]c(=N)s1)=O c1(C(=O)NC2(C3N(C(C(C(C)C)C#N)=O)CCC3)CC2)ccc2nnn(C)c2n1 C1(C(=O)NCC2N(C(C(CC=C)(C)C)=O)CCC2)CC2(CCOCC2)C1 c1(C(C(=O)NC2(CC)CC2)NC(=O)C(=O)NC2CC2)c(C)cccc1Br c1(C(=O)NCCO)ccc(-n2cc(CNc3ccns3)nn2)cc1 CCC(C(=O)NCC)C(C)C.C12(C(=O)NCC(C)C(F)(F)F)CC(C(=O)OCC)(C1)C2 N1(C(c2cc(C#N)no2)=O)CCCC2CN(C(=O)CC3CC4(CC4)CO3)CCC12 CC1CCN(C(=O)C=CBr)C1CNC(=O)C(=Cc1cscn1)F C(=O)(CCCCC(F)(F)F)NCC1CCN(C(c2cnc(C)[nH]2)=O)CC1CO c1(OC)c(Cl)nc[nH]c1=NCC(C1CC1)NC(c1ccc(C(F)F)o1)=O C(=O)(C1=CCCCCC1)N1CCCC(COC)(NC(c2c[nH]c(C#N)c2)=O)C1 Cc1ccc(NCC2CC(CNC(c3cnn[nH]3)=O)CO2)c([N+](=O)[O-])c1 CCCCC(CC(=O)NCCCC(N)=O)NC(=O)CSC(F)(F)F c1(C(N2CC(CNC(COC)=O)C(C)(C)CC2)=O)ccc2ncn(C3CC3)c2c1 c1(C(=O)NC(C(CO)NC(CCNC(C)=O)=O)C)ccc([N+](=O)[O-])cc1Cl C=CC(CCC)CC(=O)NC1CCC(C)N(C(=O)CCc2cnc(C3CC3)o2)C1 CC(C)(C#N)CCC(=O)N1CCCC1C(=O)NCC1(c2ccccc2)CC1(C)C N1(C(CCn2cnc(=N)[nH]2)=O)CC(NC(=O)CCC2CCOCC2)C(C2CC2)C1 CN1CCC2CCN(C(=O)CCN(C(=O)CCC3CCCCO3)CC3CC3)C2C1 c1(C(N2CC(CNC(CC(C)OC)=O)(COC)C2)=O)cc(N)cnc1Cl N1(C(CC(=O)OC(C)(C)C)=O)CCC(C)(C)C(C(N2CCC3(CCC3)C2)=O)C1 C(C1CNC1=O)NC(COC(C)=O)=O.C1(C(C)SC2CC2)CC2CCC1C2 Cc1ccc2c(c1C(=O)NCC1CCCN1C(=O)CCC1CCCO1)CCCN2 c1(C(N(CC2N(C(C(CC#C)CC#C)=O)CCC2)CC)=O)ccc2nnc(C)n2c1 C=CCC(CC(=O)NOC(c1ccncc1)C)OC(C)=O.C(=O)C1=NOCC1 C1(NC(c2nccc(CC)c2)=O)C2CCC1CC(NC(C1CC1(F)F)=O)C2 C1(CNC(c2c(C)noc2)=O)CC2(CCC2)CN1C(C1CCCC1C)=O N1(C(C2N(C(CCC=C)=O)CCOC2)=O)CC2(CCCO2)C1 CC1(C)CC(C(N2CC(F)(F)C2C2CC2)=O)CN1C(=O)C(=O)NCC(F)F N1(C(C2(C)CC(C)C2)=O)CCN(C(=O)CCc2cccc(O)c2)C(CCO)C1 CCCC(CCC)=CC(=O)N(C)Cc1cccc(CNC(=O)CCCC(C)O)c1 C1(C(=O)NC2(C(N3CCCCCCC3)=O)C(C)C2)CCCC12CCC2 C(=O)(C(C)(C)C1=CCN(C(=O)C2=COCC2)C1)NC(C=C)(C)C C(=O)(CCCCC#N)NC(CCC)C(=O)N1CCC(N2CCCC2)C1 CC1(C)CN(C(=O)C=Cc2ccccc2)CC1NC(=O)COC1COC1 CC(C(=O)N1C2CCC1CN(C(C1(C#N)CCCOC1)=O)CC2)C(C)S(C)(=O)=O c1(N2CC(N(CC=C)C)C2)cccc(Cl)c1Cl c1(C(N(C2CCN(C(C3CCCS3)=O)C2)CC)=O)oc(Br)cc1C Cc1nc(CNC(=O)OC(C)(C)C)ncc1C(=O)NCC1COC(=O)C1 Cc1nc2c(C(=O)NCC(C)(CC(C)C)NC(c3nn[nH]c3Cl)=O)ccnc2[nH]1 N1(c2ncnc3cc(C)[nH]c32)CCC2CCC(C1)N2C(c1cc(C(N)=O)cs1)=O C1(C(=O)NC(C#C)(C)C2CCC2)CCOCC1NC(C1CCCN1C=O)=O C(=O)(N=c1ncnc2[nH][nH]c(Br)c1-2)C1C(C(N2CCC3(CC2)COC3)=O)C1 N1(CC(CC(C)C)C)CCC2(CC1)COC(CNC(C1CC3CC3C1)=O)C2 c1(C(=O)NC2CN(c3ncc(OCC)cn3)CC2F)cccc(F)c1Br C(=O)(C1=C(C)CCC1)NCC(CC)NC(C1CC2CC1CC2O)=O C1(NC(C(CC)N(CC)CC)=O)COC2(C1)CN(C(c1ncnc(C)c1C)=O)C2 N1(C(C(C)=CC)=O)CC(N(C)C(C2CC2COC)=O)C(C)(C)C1 C(CC(=O)NCC=CCNC(C1CC1(F)Cl)=O)=CC Cc1cc(C(=O)NCCC2(O)CCN(C(=O)CCc3cccc(O)c3)C2)nn1C c1(C2(C)CC2)cccc(C(=O)NC2C=CCN(CCCC(=O)O)C2)c1 N1(C(C(CC#C)C2CC2)=O)CCC(N=[N+]=[N-])(C(=O)NC2CN(CCC)C2)C1 C(=O)(CCC(CF)CF)N(CCC(=O)NC)CC.C12CCN(C1)CCCO2 N1(CCC(N2CC(NCC(CNC(CCC#C)=O)(C)C)C2)=O)C(C)CCCC1C C(C(C(=O)N(CCC(=O)NCC(O)CC(=O)NC)OC)C(C)C)OC C(=O)(C(C)Cn1ccnc1)NCCC(C)NC(c1ocnc1C1CCC1)=O N1(CC(=O)NCC(CC)NC(c2c(C)ncn(C)c2=O)=O)C(=O)C(C)C(C)C1=O c1(C(=O)NCCC(C)(C)NC(C2N(C)CCC2)=O)ccc(F)c2c1CCC2 c1ccc(C2CC(C3CC3)C2)cc1.c1(C2(N)CC2)nnnn1-c1ccoc1 N1(C(C(C(C)C)c2cnc(C)s2)=O)CC(OC(C)(C)C)CC(C)C1 c1(C(N(C(C=Cc2n(CC)ccn2)=O)C2CC2)=O)ccc(C)nc1NC CP(C)(=O)c1csc(=NCCOc2ccccc2NC2CCC2)[nH]1 N1(C(C(CC)OC2CCCC2)=O)CCC2(CC(NC(C3CCC=CO3)=O)CO2)C1 c1(C(C)C)c(NC(=O)N(C)Cc2ccnnc2)cnn1-c1ccccc1 c1(NCCCOC(CSCCC)=O)cc(Cl)c(Cl)cc1O C1(NC(C(CC)n2cccn2)=O)CN(C(c2cc(C)c(F)cn2)=O)CC1C1CC1 c1(C(N(CC(O)CNC(c2c[nH]ccc2=N)=O)C)=O)nc2n(c1Br)CCC2 c1(CC(N2C(CNC(C(F)=CCC)=O)C(C)CC2)=O)cccc(Br)c1C Cc1c(NC(C2CCC2CNC(c2c[nH]c(C(N)=O)c2)=O)=O)cccc1F CC1=NN(c2cc(C)ccc2C)C(=O)C1C(=O)OCCOC1CCO1 c1(OC)cc(CC(=O)NC2CC(NC(c3occc3C)=O)C2)cc(Br)c1 CCC(CC(=O)N1CC2(CC2)CC1C(=O)NC1CCCSCC1)C(F)F c1(C(N2CCCC(CCNC(c3cc(C)n(C)c3)=O)C2)=O)ncc2ccccn12 c1(OC)ccc(N)cc1C(N1CCCOCC1C)=O N1(C(C(C2CC2)NC(CCN(CC)CC)=O)=O)CC2(CSC2)C1 c1(C(=O)NCC2(O)CCN(C(CC3(C)CCC3)=O)C2)sc2cccnc2c1Cl C(CN=[N+]=[N-])(C(=O)NCC(C)(C)C(F)(F)F)NC(c1n(CCC)ccc1)=O N1(C(C(C(C)O)C)=O)CCCC(C2CN(C(c3ccc4ncccc4n3)=O)C2)C1 Cc1[nH]nc2c1CC(C(N1CC3CN(C(c4ccsc4Cl)=O)CC3(C)C1)=O)CC2 C1(C2(NC(=O)Cc3ccsn3)CC2)CCCN1C(C1CCSCC1)=O C1(C(N2CC(C(C)NC(COCCSC)=O)C2)=O)CC12CC(C)(C)C2 CC1CCCN(C(C2CC3CCCC23)=O)C1CNC(=O)COC1COC1 c1(C(C(=O)NCC2C(NC(CSCCCC)=O)CC2)C)ccccc1F C1(CC(=O)N(C(COC)C)C)C2CN(C(C3CC(COC)C3)=O)CC12 C(=O)(CC(C(C)CC)NC(c1ccc(C#N)c(C)c1)=O)NC(C(C(=O)OC)C)C C1(NC(c2cnc[nH]2)=O)CN(C(=O)CCCn2cccn2)CC12CC2 CC1(C)C(CN(C2CCCC2)CCCOC2CCC2)C1(C)C C1(O)(C(N2CCC(N(C)C(c3ccnn(C)c3=O)=O)C2)=O)CCCC(C)(C)CC1 C(C(C(=O)OC)C(C)(C)C)OCCN(C(=O)C(=O)NCCC(=O)OC)CC c1(C(=O)Nc2ccc(NC(C(OC)OC)=O)cc2)cc2cccnc2[nH]1 Cc1cccn(CC(=O)NC23CC(NC(C4C(F)(F)C45CCC5)=O)(C2)C3)c1=O C12(C(=O)NC(C3CCCN3C(=O)C(CO)N(C)C)C)CC(C)(C1)OC2(C)C C(=O)(CCC(=O)c1cnn(C)c1)N(CC(CN(C(C=CC(CC)C)=O)C)O)C c1(CN(C(=O)CC2(C)CN(Cc3ncc(CN)o3)C2)C(C)=O)cnc(Cl)cc1Br Cc1cnn(C)c1-c1cn(CC2CCN(C(c3cnc(C4CC4)s3)=O)C2)nn1 c1(-c2nc(C3C(O)CCC3)n(C3CCC3)n2)ccc(Cl)cc1O N1(C(C2ON=C(CC)C2)=O)CCC(F)(C(=O)NCCSCC(=O)OC)CC1 C1(CC)CN(C(=O)CCOC2CN(C(=O)CCn3cc(C)cn3)C2)CC(=O)N1 C1(CC)OCCCC1C(=O)NCCCOCCNC(=O)CCCN(C)C CN1N=C(CC(=O)NC2CC3(C2)CC(CNC(c2cc(C#N)c[nH]2)=O)C3)CC1=O N1(C(C2(NC(C3CCCOCC3)=O)CCC2)=O)CCCC(OCC)(CO)C1 C#CC1(O)CCCN(C(c2ccc(CNC(=O)CCCN(C)C)s2)=O)C1 c1(N2CC(CSC(F)(F)F)C2)cccc(C(F)(F)F)n1 C1(NC(=O)NCC(c2ccc3c(c2)OCO3)OC)CCOC12CCCCC2 Cc1ncc(C(N2CCC2CC(=O)NCCC2CSCCN2)=O)n1C O=C(C1=NOC2COCC12)NC1(C(N2CC(C3CC3(F)F)C2)=O)CC(F)(F)C1 S(=O)(=O)(CC(=O)NCCC1(CNC(=O)CCn2cc(C)cn2)CC1)N(C)CC c1(N2CCC(CC=C)(NC(C3CC3(C)CC)=O)C2)ncn(C)c(=O)c1Br c1(C(N2CC3C(CNC(Cc4cc(C)no4)=O)(C3)C2)=O)c[nH]c2ncc(F)cc12 N1(C(c2[nH]cc(C)c2C)=O)CCOCC12CCN(C(c1cnoc1)=O)C2 c1(C(=O)NCC=CCNC(C(C(CC)O)(C)C)=O)c[nH]c2ccc(C#N)cc12 Cc1c(C(N2CC(C(=O)NOCC(C)(C)O)CC(C)C2)=O)cccc1F C1(NC(C=C(C)C(F)F)=O)CCN(C(=O)C(F)C(F)(F)F)CC1(C)C C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C)N(C(=O)COC2CCCC(C)C2)CC1 C1(CNc2cccc(C3(C)NC(=O)NC3=O)c2)CCC2(CCC2)C1O Cc1cc2[nH]c(C(=O)NC(C)(C)C(C)NC(=O)Cc3nnc(C)o3)cc2o1 c1(C(=O)NCC2CCCN2C(c2cccc(OCC)c2)=O)nccnc1Cl.CC#N c1(NC(CC)C2CC2)ncc(C)cc1S(=O)(=O)NCC1CCS(=O)(=O)C1 c1(C(=O)NC(C(C)(C)NC(C2C(C(=O)OC)CC2)=O)C)cc2ccccc2cn1 Cc1ccc(C)c(C(=O)CCC(=O)NC2CCC2NC(c2nnsc2C)=O)c1 N1(C(c2ncc(OCC)nc2)=O)CCC2CN(C(c3cc(C)ncn3)=O)CC2C1 C(C(C)(O)CC(=O)NCC1(C(N2CCCC(C)C2C)=O)CCCCC1)OC C(=O)(C(C)(C)C(F)(F)F)N1CCC(CN(C)Cc2ccc(C)cn2)C1 c1(NC(c2c(OCCCC(=O)OC)cccc2)=O)cc(=O)n(C)cc1Br Cc1oc(OC(C2(NC(=O)OC(C)(C)C)CCCC2(C)C)=O)c(C#N)c1C c1(CCC(=O)NCC(F)CSC)nccn1C.C(C(=O)NCCO)N(CC)CC c1(C(N2C(c3cn(CC(CC)O)nn3)CC2)=O)ccc(F)c(C)c1 c1(C(=O)NCCSCc2ccccc2)cc2c(cc1F)NCCC2 C(=O)(C1=CCC(C)(C)CC1)NCC(C(C)C(C)C)NC(CCC1CC(OC)C1)=O N1(C(COC(C)=O)=O)CCCC(C(N2CCC(CN(C)C)C2)=O)CC1 c1(C(C)=O)ccc(N(C)Cc2cncn2C)cc1 N12CCCC1C=CC2=O.C1(NCc2ccc(CC)o2)CCCC(C)C1 CN1C(=O)NCC1C(=O)NCC1CCC(NC(c2nccnc2C(N)=O)=O)CC1 c1(OCC)cccc(Cl)c1C1CC1C(=O)OCc1csc(CC(C)C)n1 C1(CC(N2CC(SC)C2)=O)CC2(C1)CN(C(c1ccc(CO)o1)=O)C2 c1(C(=O)NC2CCC(NC(c3cnc(CC4CC4)s3)=O)C2)cnn2cccnc12 c1(C(N2C(C(C)(C)NC(=O)COc3ccsn3)CCCC2)=O)cccc(Cl)c1F c1(CSC)cccc(CCNC(CC2(N(C(c3cccnc3)=O)C)CC2)=O)n1 Cc1cc(NC2CN(C(c3csc(CC(C)C)n3)=O)C2)n2ncnc2n1 C12(C(N3CCC(NC(c4c(C)occ4)=O)CC3C3CC3)=O)CC(C3CCCC3)(C1)C2 c1(C(N(CC(C)CNC(C2CC2C)=O)C)=O)ccc([N+](=O)[O-])cc1Br C(CCC(=O)NCC(C)NC(=O)CC1CCOC1C)OCCOCC c1(C(=O)Nc2c(C)ccc(OC)c2)cc2cc(-c3cncn3C)ccn2n1 c1(CC(N2CCC(N(C(C=CC)=O)CC)C2)=O)ncccc1F N1(C(c2c(OC)nsc2)=O)CCC(C)C1C(=O)NC(CN(C)C)CO N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(c2ccc(CF)cc2)=O)C(C)C1C C1(NCCNC(c2ncc(Cl)cc2Cl)=O)CCS(=O)(=O)C2(C1)CC(CO)C2 c1(COCC(=O)NCC(=O)N)nc(CO)cs1.C(C(C)(C)CN(C)C)N(C(C)=O)CC C(=O)C1c2c[nH]nc2CN1.c1(C(=O)O)ccc(CC2CN3CCC2C3)o1 C1(CNC(c2n(CC=C)nnn2)c2csc(C)c2)CC1C1CCC1 c1(-c2nc(Cc3cc(OCC)ncc3)nn2C)cn2nc(C(F)(F)F)ccc2n1 C(CC(C)OC(C)C)CNC(C1(NC(C(C)OC(C)=O)=O)CCCC1)=O C(=O)(C(F)C(C)(C)O)NCCCCN(C)C(c1csc([N+](=O)[O-])c1)=O c1(OC)ccc(CN2CCC3(CC3C(=O)Nc3cn(C(C)(C)C)cn3)C2)cc1Br CCCC(C)(C)C(=O)N1CC(C(C)N(C2CCOC2C)C)C1.C1C(=O)N1 C(=O)(C(F)(F)CC1CC1)N(CCCN(C(C(COC)N(C)C)=O)C)C n1(CC)cnc2c(NC(C)CN(C)Cc3cncn3C)ncnc12 CC1CN(C(c2cnc(S)nc2)=O)CCN1C(=O)CCC1CC(C)(C)CO1 c1(C(=O)NC2C(Nc3nccc(OC)n3)CCCC2)cc2nnn(C)c2s1 Cn1nc(C(=O)NCCC2(CNC(C3CCC(C)O3)=O)CC2)cc1C1(Cl)CC1 C1(CC)C(NC(c2cccnc2O)=O)CCCN1C(=O)CC1CCC2(CC1)CC2 c1(OC)c(C(C(=O)NCCN2CCOCC2)NC2CCCC2C#N)cccc1Br C(=O)(C1=CS(=O)(=O)CCC1)NC1CC(CNC(C=C(C)c2ccco2)=O)CC1O c1(CNCC(c2ccc(C)o2)O)ccc2c(c1)C(=O)N(C)C2 CC1(C)CCCC(CC(=O)Nc2cccc(NC(=O)CC(=O)NC3CC3)c2)CC1 Cc1cccc(C2(C(N3C(CC4(CBr)CCOCC4)CCC3)=O)CCC2)c1 Cc1cncc(C(=O)N(CCN(C(=O)C2=CCCC2)CC)Cc2ccccc2)c1C CCCC(C(=O)N1CC(CNC(c2cc(C(=O)NCCO)cs2)=O)C1)OC CC(C)CCC(C(=O)N1CC(O)(CO)C1)NC(=O)CCN(C)C N1(C(CCCCC)=O)CC(C(N2CC(n3ccnc3)C2)=O)CC12CCC2 C1(C(C)NC(c2c(CC)nc(C)s2)=O)COc2ccccc2O1 c1(C(N2CCC(NC(C3C(C)C3)=O)C2)=O)ccnc(Cl)c1Cl Cc1nn(C)c(C(F)F)c1C(=O)NCC1(O)CN(C(=O)C(C)CC2CC2)C1 c1(C(C(N2CCC(N(C(=O)CCC3CC3(C)C)CC)C2)=O)O)ccccc1CO CCCCCCCCC(=O)N1CCC2(C1)CN(C(C1(CF)CCC1)=O)C2 c1(C(N(CC(C)NC(c2nn(CC)c(C)c2)=O)C)=O)cc(Cl)cnc1OC CC(C(c1nnnn1Cc1cccs1)NCC1C(C)(C)C1(C)C)C(C)(C)C N1(C(C2CC23CC3)=O)CC(NC(C23CC(C2)C3)=O)CC2(CCC2)C1 C(C(C(=O)NCC12CCCC1CCC2)C(C)C)NC(c1c(C)cnnc1)=O c1(C(N2CC(O)(C(CNC(C(C)=C3CC3)=O)(C)C)C2)=O)cc(C(N)=O)cn1C c1(N2CCC(NC(CC)=O)CC2)cc(NCC2(C)CC(C)C2)nc(C(C)C)n1 Cc1nn(C)c(C(=O)NC2CCCN(C(c3cccc[n+]3[O-])=O)C2C)c1Br N(C(=NCCF)N(C)CC12CCC(F)(CO1)C2)N(CC(=C)C)Cc1ccccc1 CCCCCC(F)C(=O)NC(C)C(=O)NC1CC(N(C)C)C1 c1(OC)ccc2c(c1)OCC(C(N1CCC(NC(C3(O)CCOC3)=O)C1C)=O)C2 N#Cc1c[nH]c2ncnc(N3CCC(N4CCOCC4)C(O)C3)c12 CC1CCC=C1C(=O)N1CCN(C(c2ccncc2)=O)CC1c1cccnc1 c1(C(N2C(COC)CN(C(=O)C3=NNC(=O)C3)CC2)=O)ccc2c(c1)ncn2C Cc1cc(F)c(C(N2CC3CCC3(NC(=O)C#CC(C)C)C2)=O)cc1F c1(C(=O)NC2CCC(CNC(C3(OC)CC(OC)C3)=O)CC2)c[nH]c2ncccc12 N1(C(C(C)(C)CF)=O)CCC(C=CC(=O)NCCc2ccns2)CC1 CC1CC2C(CC(OC(c3nc4cc(N(C)C)ccc4[nH]3)=O)N2OC(C)=O)O1 CC1(C)Cc2cccc(C(=O)NC3CCCC3CNC(=O)CCCC3CC3)c2O1 Cc1ccccc1S(C)(=O)=NC(=O)c1sc(Cl)cc1CC#N c1(C(c2n(C(CC)C)nnn2)NCC2(C)CSC2)cc(S(C)(=O)=O)ccc1F c1(CNC(CCNS(CC)(=O)=O)=O)nc(NC(C2CCCN2C(C)C)=O)cs1 Cn1ccc2cccc(C(=O)NC3CC3C(=O)Nc3ncc(Cl)nc3Cl)c12 C1(OC)CN(c2nc(NCc3ccc[nH]3)c3c(ncn3C)n2)C2(CCOCC2)C1 C1(Cl)(C(N(CCNC(=O)Cn2cc(C3CCC3)nn2)CC)=O)CCCCC1 N1(C(=O)OC)CCCN(C(C2CNC(=O)N2C=C(Cl)Cl)=O)C(C)C1 C1(C)(C(=O)NC2C3CN(C(c4c(O)ccc(OC)c4)=O)CC32)CCC(F)(F)CC1 c1(C(=O)NC2CCN(C(c3c[nH]cc(C)c3=O)=O)C2)cc(S(N)(=O)=O)ccc1O N1(C(CC(C)(C)C)=O)CC(C(=O)NCCNC(=O)C2CC2)C2(CC2)C1 c1(C(=O)NCC2CN(C(C3(C=C)CCC3)=O)CC2C)cc(Cl)ccc1F c1(C(=O)NC2CCN(C(=O)C(F)(F)CO)CC2F)cccc2cncn12 C1(C(=O)NCC(N(C)C(c2cc(C(F)F)nn2C)=O)C2CC2)CN(C)CCN1C CC(C(=O)NOCc1cn(-c2ccc(F)cc2F)nn1)C(C)(C)C C1(C(N2CC(CCCCNC(Cc3c(C)oc(Cl)n3)=O)C2)=O)C2(CCC2)C12CCC2 C(=O)(N=c1cc(Cl)n(C)[nH]1)N1C2CCN(C(C(COC)(C)C)=O)C2CC1 C(=O)(CC(C(F)F)NC(C1CC2(CCO1)CC2)=O)NCCC=CCCC Cc1ccc(C(C(=O)NC2(CCNC(C3CC3[N+](=O)[O-])=O)CC2)C2CC2)cc1 N1(C(=O)NCCc2ncc(SC)s2)CCC(O)CC12CC2 c1(C(N2CCC(N(C)C(C3CCC(C)(C)C3)=O)CC2)=O)nc2cc(O)ccc2[nH]1 Cc1ccc(C)c(C(=O)NC2CCCC2NC(c2nn(C)c(Cl)c2Cl)=O)c1C C1(COC)CN(C(c2csc(CNC(=O)C(C)c3ccsc3)c2)=O)C1(C)C N1(C(=O)C2=NOCC2)CC2(CCN2C(c2cc(O)ccc2Br)=O)C1 c1(C(=O)NC2CCN(C(C3N(CC)CC3)=O)C2C)ccc2nc(O)oc2c1 C1(c2n(C)ncc2)CN(C(c2cnsc2)=O)CC1NC(=O)CC1CCC=CCC1 CC1C2C(CCN2C(c2cc([N+](=O)[O-])ccn2)=O)CN1C(=O)C(O)C(C)(C)C C#CCC(C)C(=O)NCC1C2CN(C(C3CCC(C(F)F)CC3)=O)CC12 Cc1cc[nH]c1C(=O)NCC1COC(CNC(C2CCC2CN(C)C)=O)C1 C(=O)(C1=CCSC1)N1CC(O)(CN(C)C(c2cccc(Cl)c2)=O)C1 C1(NC(CSC(C)C)=O)COC2(CCCN(C(c3cc(N)c(F)cc3F)=O)C2)C1 c1(NC(CCOC)COC)cc(N(C)CC2CN(C)CCO2)nc(C)n1 N1(C(C2C(CC(C)(C)C)C2)=O)CC2CC(C(=O)NC(C3CCCO3)CO)CC2C1 c1(C(N(CCCNC(c2nn(C)c(Cl)c2Cl)=O)C)=O)coc2c(F)c(Cl)ccc12 C1(O)(CCNC(CCSC)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1 c1(-c2nc(C(CC)CC)nn2-c2ccc(C)cc2Cl)cc(C)nc2c1CCCC2 CC12CN(C(=O)CC3CCCO3)C(C(=O)NC3CC3C3CCC3)(C1)C2 c1(CC(=O)N(CC(CNC(C(C)CN(C)C)=O)O)C)cc2cc(Cl)ccc2[nH]1 c1(C(N2CC(CCC(=O)OCCOC)C(=O)CC2)=O)nccn2cnnc12 C1(N(C)C)CCC(NC(C23CC2CCN3C(c2cc(C(N)=O)c[nH]2)=O)=O)CC1 C(C)(C)(CCCNC(c1cnn(CC2CC2)c1)=O)NC(C(F)=C(C)C)=O C1(C(=O)NCC(CC)C)CCN(C(=O)Cc2cncn2C)CC1(C)C CCCC(C)CCCC(=O)Nc1ccsc1.C1CCN(C)CCCNC(=O)CO1 c1(OC)cccc(CN2CCCC(NC(=O)CCN3CCOC3=O)C2)c1 N1(C(C2(CC=C)CCC2)=O)CCC(NC(c2ncsc2C)=O)C(CO)CC1 c1(C(C)NC(c2nnnn2CC2CC2)CCCC)nnc2n1CCC2.O c1(CC)cccc(C(N2CC3CC3(CNC(=O)COC3CC(F)(F)C3)C2)=O)c1O C1(C(=O)NCCCCOCC)CCCC1NC(=O)CC(=O)N(C)C C1(NC(C(COC)OC)=O)CCCC12CCN(c1ccnc(C#N)n1)CC2 C12(C(N(C)CCC3CCC3)=O)CCCC1CCN2CC=CC(F)(F)F Cc1ncc([N+](=O)[O-])n1CC(N1CCC(C)(C)C1CNC(c1ccsn1)=O)=O C1(NC(C(CC)N2CCCC2=O)=O)CN(C(C2CC(C)C2)=O)C2(CCOCC2)C1 C1(C)(NC(C(CCC)NC(N2CC(OC)C2)=O)=O)CC1(Cl)Cl.C12CN(C1)C2=O.OC c1(CC(=O)NC(CCN(C)C(C2CC2(C)C(F)(F)F)=O)C)nc(O)n[nH]1 c1(-c2c(C3CN(C)CC4(CC4)C3)ccc(F)c2)cc2nc(OC)ccc2[nH]1.OC CC1(C)CC(CNC(=O)C=CCO)N(c2cncc(C#N)n2)C1 c1(C(N2C(CNC(C3C(CC(C)C)C3)=O)CCC2)=O)cc(Cl)c(N)cc1F c1(CN2C(C(=O)Nc3ccc(Cl)nc3I)COCC2)cc(F)c(I)c(F)c1 CS(=O)c1ccc(C(N2CCCCC(NC(c3cc(O)cc(O)c3)=O)C2)=O)cc1 c1(OC)ccc(CN2CC3(CC(CC(N4CCC(C#N)CC4)=O)C3)C2)cc1C C1(C2CCN(C(c3n[nH]cc3Br)=O)C2)(NC(c2nnn3c2CSCC3)=O)CC1 c1(CC)cc(C(N2CCCC2(C)C(=O)NC(C2CCOCC2)C)=O)ccc1F c1(CC)ncc(C(=O)NC(CCN(C)C(c2nn(C)cc2C)=O)C(C)C)c(O)n1 CC1CN(C(=O)CCCn2cc(C3CC3)nn2)CC(C)N1Cc1cccc(F)c1 c1(NC(C(C)OC(C)(C)C)=O)cccc(C(=O)N(CCO)CC2CCOCC2)c1 c1(C(N2CCC(OC)(CNC(C3CC(O)(C#N)C3)=O)C2)=O)cc(C)cc(C)c1O CCC1=C(C(=O)NCC2CN(C(=O)CCC(C)SC)CCO2)SCCO1 c1(C(C)C)ccc(-c2nc(Cc3ccc(Br)cc3)n(CSc3cccs3)n2)cn1 C1(N(C(C(c2c(C)noc2C)C)=O)C)CCCN(C(C2CC2C(C)O)=O)CC1 c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)C(c2cc(C)oc2C)C)C3)cc1 C(=O)(C(CC(C)(C)C)OC)N1CC(CC)N(C(c2cc(C3CC3)on2)=O)CC1 C1(CCNC(C(CC)=CCCC)=O)CN(C(C2(C(N)=O)CCC2)=O)CC1C C1(N(C(=O)CC2(C)CCC2)C)CN(C(c2ncnc(O)c2F)=O)CCC1O N1(C(c2n(C)cc(I)c2)C(=O)NCC2CC2)CCC(Cn2cncn2)C(F)(F)C1 CN1CC2C(C(=O)NC(c3nocc3C(=O)NC3(C)CCOCC3)C)C2C1 C1(CN(C(C(N2CCOC2=O)C)=O)C)CCCN1N(C)C(c1ccc(CO)s1)=O C=CC1CCCCN1C(C1CC(C)(C)CN1C(=O)C(CC)n1ccnc1)=O c1(CC(=O)NC2CCC(CCNC(C(F)=CC)=O)C2)cccc(SCC)c1 C(=O)(C(C)(C)n1cc(Br)cn1)N(C)CC1(N(C(=O)CC2(C(=O)OC)CC2)C)CC1 c1(N(C(C)C)C)ccc(C(=O)N(CC(O)CN(C(=O)C(C)C2CC2)C)C)cc1 C1(C(C)NC(=O)C=CCO)CN(C(=O)CCc2nc(-c3ccsc3)no2)CCO1 c1(C(=O)OC)cnn2c(-c3ccc(N4CCC(n5ccnn5)CC4)cc3)ccnc12 c1(COC)ccc(C)c(C)c1.c12ccc(s1)[nH]c2=O.C1C(N(C)C)C(=O)N1 N1(C(C(C)OC)=O)CC2CC(C(N3CCCC(F)C3)=O)(C2)C1 C1(C(=O)NC2CN(C(c3n4c(nn3)SC(=C)C4)=O)C2)CCOC2(CCOCC2)C1 C(CN=C(NCC(C)C)NC(c1ccn(C)n1)C)c1c(C)nn(C)c1 N1(C(C2C(=C)C2)=O)CCC(CCNC(=O)Cn2ccc(C(F)(F)F)n2)C1 C[S+](C)CCC(O)C(=O)N1CCN(C(c2ncccn2)=O)C(CC(F)(F)F)C1 c1(C(=O)NC(C2CCCN2C(C2(C(F)F)CC2)=O)C)nn2cccnc2c1Cl C1(C(=O)NCC2CCN(C(C(C)C3CC3)=O)C2)CCCNS1(=O)=O C1(C)(C(N(CCN(C(c2cc(C)ncn2)=O)CC)CC)=O)CCCC1O CC(C)(CNC(C1(C)CCCS1)=O)CCNC(C1C(C(F)(F)F)C1[N+](=O)[O-])=O c1(N(C(C)=O)C(C2C(C)C2C)=O)cccc(C(=O)N(C2CCCC2)CC#N)n1 C1(CNC(COCCNC(c2c(C)cns2)=O)=O)OC(=O)CC1(C)C C1(C(N2CC(COC)(NC(=O)C3=CCCCC3)C2)=O)CCCC(C)(C)CC1 C1(NC(c2c(C)oc(C3CC3)c2)=O)CCN(C(=O)CSC(F)(F)F)C(C)C1 c1(C(N2CC(NC(c3c(C)nc[nH]3)=O)C(C)C2)=O)cc(C(F)(F)F)ccc1O n1(CC)ncc(C(=O)NCC2C(CNC(=O)C=Cc3cscn3)C2(F)F)n1 C1(NC(CSCC(C)C)=O)CCC2(CC1)CCN(C(C1CCC(=O)CC1C)=O)C2 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCCN(C(CCCOCCC)=O)CC1C C#CCCCCCCC(=O)N(C(C)CNC(c1cccc(-n2cccn2)n1)=O)C C1(CC(=O)N(CC(c2ccccc2)NC(=O)Cc2csnn2)CC)COCCN1C N(C1CCC(CCC(c2cccc([N+](=O)[O-])c2)C)c2ccccc21)Cc1ccc(Cl)cc1.n1(CC)nnnc1 C(C(C)CC(=O)NC1CCCC1O)NC(c1cnc(C)o1)=O N1(C(CCCn2cnnn2)=O)CCOCC1CO.c12cc[nH]c1C(=O)NC2 N1(C(c2cncc(OC(C)C)c2)=O)CC(NC(=O)CCn2ccnn2)CC1(C)C C(N=c1nc2c(ncn2C(C)C)c(NCc2cccc(N)c2F)[nH]1)c1c(C)ccs1 C#CCCCCCCN(C(C1(CC=C)CCN(C(=O)C2=CC(C)(CC)C2)C1)=O)CC c1(C(N2C3CC(C(N(CCCCCC=C)C)=O)(OC3)C2)=O)ccc2nn[nH]c2c1 CCCCC(F)C(=O)N1C2CCC(C2)C1CCNC(=O)CC(=O)NCC c1(OC)ccc(C)c(C(=O)N(C)CCNC(=O)C(C)C2CCCO2)n1 Cc1nc2c(N3CCC(OCCNC(=O)C(C)(C)C(F)(F)F)C3)ncnc2s1 c1(C(=O)NCC(C)N(C(c2ccc(O)cn2)=O)CC)ccc(C)c(Cl)c1Cl C(CC(C(=O)N1CC2CC1(CNC(C1CCC1)=O)C2)NC(c1ccco1)=O)SC c1(C(N(C2CCN(C(CC(C=C)C)=O)C2)CCO)=O)cccc([N+](=O)[O-])c1 c1(C(N(CCCNC(C2CN(C)C2)=O)CC)=O)cccc(SCC#N)c1 C(=O)(CCCC(F)(F)F)N1CC(C)C(CNC(=O)CSCCN2CCCCC2)C1 C1(C(N2CCC(C(=O)Nc3ncc(F)s3)C2)=O)CCC(F)(F)CC1 N1(C(c2c(C)nncc2)=O)CCC12CN(C(C1(C)CC1(C)C)=O)C2 N1(C(c2ncc(OCCOCC)nc2)=O)CCC(CCOC)CC1C c1(CNC(C(=O)NCC2(C)CCCC2(F)F)=O)nnc2n1CCCC2 Cc1cccc(C(N2CCCC(CN(C(C34CCCC3C4)=O)C3CC3)C2)=O)c1Cl N1(C(=O)NC(c2c(C)nccn2)C)C2CCC1C(COc1c(C)cccc1C)C2 C(CC(C(C)C)NC(c1cnc(C(F)(F)F)cn1)=O)NC(CNC(C)=O)=O N1(C(CCC(C)C)=O)C2CCC1CC(CNC(c1ccc([N+](=O)[O-])s1)=O)C2 C=C(C)C1OCCC1C(=O)NCC1(C)CCN(C(=O)Cc2nnc(O)s2)CC1 c1(CC)cc(C(=O)NC(CO)C(C)NC(c2cc(Br)cn2C)=O)c(C)nn1 C1(CNC(c2cc(C(C)C)[nH]n2)=O)CCN(C(=O)CCC2CCC(=O)N2)C1(C)C c1(C(=O)NC(CNC(C(C=C)O)=O)(C)Cn2cccn2)cccc(Cl)c1O C(c1ccccn1)=CC(=O)NCCCC(C)NC(c1n(COC)ncc1)=O C=CCC(C)(C)C(=O)NCCCCN(C)C(c1ccc(C(F)(F)F)s1)=O c1(OCC)ccccc1NC(=O)C(C1CCN(C(c2cccnc2C)C)CC1)C c1(C(N(CCCNC(C2(C)CCCNC2=O)=O)CC)=O)ccc(C#N)cc1O c1(CC)ccc(CCNC(N2CCCC(c3ccc(C(C)C)cc3)C2)=O)cc1 C1(C(=O)OC)C2=CC(CC2)C1C(=O)Nc1cnc(-c2ccsc2)s1 C1(C(N(C)CCN(C)C(C2CCCNS2(=O)=O)=O)=O)CN(CP(C)(C)=O)C1 c1(C(=O)NCC(CNC(c2c(C)ncnc2O)=O)O)ccc2nc[nH]c2n1 C(=O)(C(CC(F)F)NC(=O)CC1CC2(CC2)CO1)NCc1occ(C)n1 C(C)(CCN=c1[nH]c(=NC2CCn3nnnc3C2)c2c(F)cccc2[nH]1)SC c1(C(=O)NCC(C)N(C(c2c(C)nns2)=O)C)cc2c(cc1F)NCCC2 N1(C(CNC(C(CC)CC)=O)=O)CCOCC(CNC(C2CC2F)=O)C1 CC(CC(C)(c1nnnn1C1CCCC1)NCCF)C(F)F.C12CC(C1)NC(=O)C2 C1(C(N2CCCC(OCC)C2)=O)CN(C(c2ccnc(CO)c2)=O)CCC1(C)C C1(CCC(=O)NC2(C)CN(C(c3cnn(CC)n3)=O)C2)CCCC(O)C1 c1(-c2n(-c3ccc(CCOCC)cc3)nc(COC)n2)cc(Br)cnc1CC N1(C(CC(CNC(=O)COC(F)(F)F)OC)=O)CC2(C1)CC(C)(C)C2 Nc1c(Cl)ccc(C(N2CC(NC(=O)Cc3cccnn3)C2)=O)c1Cl c1(CCNC(C2CNCC2F)=O)cc2cnccc2[nH]1 c1(C(C(=O)N(c2ccccc2SC)C)N(CCCCCC)C)ccc(F)cc1C c1(C(=O)NCC(C2CC2)OC)coc(CNC(=O)C(C)(C)C2CCOCC2)c1 Cc1cc(NC(C(=O)C(C)(F)CC2CCCC2)=O)ccc1O.C1(N)CCOCC1 N1(C(c2c(OC)scc2)=O)CC(NC(C2CCCOC2C)=O)C(C)C1 Cc1ccc(C(CO)NC(=O)C(=O)Nc2csc(-c3ccc(Cl)cc3)c2)cc1 C(=O)(CCS(=O)(=O)C(F)(F)F)NC1CC(CNC(C(COC)O)=O)C(O)C1 N1(C(C2CN(CC)C(=O)C2)=O)CC(C(=O)NC(C2CCCC2)C)CC(C)(C)C1 c1(C(N(C(C)CCNC(=O)Cc2ccco2)C)=O)nccc2cnn(C)c12 C1(CNC(C=CCCC(C)C)=O)CCCN(C(=O)C(C(C)C)c2ccccc2)C1 Cc1cc(C(=O)C(C)NC(=N)O)c(C)n1-c1nccs1.c1(CC(=O)O)ncnn1C c1(C(=O)NC2CC(CNC(C3C=CCCC3)=O)C2)ccc2c(Br)cnn2c1 N1(C(c2[nH]c(=NC)sc2)=O)CCC2(CC1)C(OC)CC2NC(=O)CNC=O N1(C(CN(C(CCC)=O)CC(F)F)=O)CCC(NC(=O)C(F)(F)F)CC1 Cc1nn(C)c2c(NCCS(N)(=O)=O)nc(=NC3COc4c(F)cc(F)cc43)[nH]c12 N1(C(c2cc(CCC)nn2C)=O)CCC(O)(C(C)NC(=O)CSC(F)F)CC1 C1(NC(C(C)(C)Cl)=O)CCN(C(=O)COC2CC=CC2)CC1O C(COC)(C(C)(C)C)NC(c1n(CCCOC)nnn1)c1occc1C(C)C C#CC1(CNC(=O)CC2CCC(NC(c3sccc3Cl)=O)CC2)CCCC1 CCC(C(=O)NC(C(=O)O)C1(C)CC1)n1ccc(-c2ccccc2)n1 Cc1nn(CC(=O)NCCOc2cccc[n+]2[O-])c2ccccc12 c1(SC2(C(c3nnnn3C3CC3)NC3(CS(C)(=O)=O)CCC3)CC2)ccc(Br)cc1 C1(NC(Cc2c(C)non2)=O)CCC(C)N(C(c2ccc(C(F)F)o2)=O)C1 C(C(C)C(=O)NCCO)NC(CCN(C(CCC)C)C)=O C1(C(=O)NCC(CSC)(C)O)C=CCN(C(=O)CC23CCC(CC2)C3)C1 N1(C(c2c(C)cc[nH]c2=N)=O)CCN(C(c2cnc(C(F)F)s2)=O)C(C)CC1C C(N=c1[nH]nc(C2CC2)o1)C1C(NC(Cc2c(OC(C)C)cccc2)=O)CCC1 N1(C(CN(C(=O)CC2CCOC2(C)C)CC)=O)CCC(F)(F)C(F)C1 C1(C(N2CCC(CNC(CCCc3cc(C)no3)=O)C2)=O)CCC2C1C2(F)F Cc1nc2cc(C(=O)N(C3CC4CNC3C4)CC3CC3)ccc2s1 C1(NC(CC(=O)NCC#C)=O)CCC12CCN(C(c1cnn(C)c1N)=O)CC2 c1(CC)nnc2n1CCCC2C(=O)NC1(CNC(=O)C(F)n2cccn2)CCCC1 C1(C(N2CC(CNC(C3(CC#C)CCOC3)=O)C2)=O)CC2CC(=O)C1C2 N#Cc1ccc(SCCC(N2CC3(CNC(C4CC45CC5)=O)CCC2C3)=O)cc1 C1(C(N2CCC(CN(C)CC3CCCC3)C2)=O)(CC)CCCN(C(=O)COC)C1 C1(C)(C(=O)NCCCN(C)C(C2(Cc3ccccc3F)CC2)=O)CCCCC1 N1(C(C#CC)=O)CC2(CC2)CC1C(=O)NCC(O)Cc1ccc(F)cc1 C1(NC(c2c(CC)cno2)=O)CCCC(NC(=O)C(C2CCOCC2)C)C1 c1(C(N(C)CCOCCCN(C)C(C2(N=[N+]=[N-])CC2)=O)=O)cccc(CO)c1 C12CCN(CC1)Cc1cn2nn1.C1(C(=O)NCC(F)(F)CO)CC12CCC2 N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC(F)(CNC(c2ccc(Cl)o2)=O)CC1 c1(C(N(C(CCNC(CCC(C)CN(C)C)=O)C)C)=O)cnn2ccn(C)c12 Cc1ccnc(C(=O)NCC(C(C)(C)C)NC(C2(C)C=CCCC2)=O)c1 C1(C(=O)NCC2CN3CCC2C3)C=CCN(C(c2ccc(Cl)o2)=O)C1 CN1CCC(C(=O)NC(CNC(C2(C(=O)NCC3CC3)CCC2)=O)C2CC2)C1 C=C(Cl)CC(C(=O)Nc1ccc(OC)c(C)c1)NC(c1ccn(COC)n1)=O Cc1ccnc(C(=O)NC2CCC2NC(c2cncc(C(N)=O)c2)=O)c1F N1(c2c(OC)cncn2)CC(C2CCCN(C(c3ncoc3C(F)(F)F)=O)C2)C1 N1(C(C2N(C)CCC2)=O)CC2CC(NC(=O)Cc3cccc(F)c3)CC2C1 N1(C(=O)Cn2ccnc2)CC2CCC2(CC(=O)Nc2cccc(F)c2)C1 c1(C(N(CC(CNC(CCCCCC)=O)C)C)=O)ccc(F)c(N)c1F C(N=c1[nH]c(=NC2CCC(CO)C2)c2c(ncn2C)[nH]1)C1CCN(CCOC)C1 N1(C(COCc2ccc(OC)cc2)=O)CCC(NC(=O)COC(F)F)C(O)C1 c1(C(=O)NC2CC2CNC(CC=C(C)C)C(=O)O)ccc2cncn2c1 C=CC(C)(C)C(=O)N1CC(CN(C(=O)NC2(CC(F)F)CC2)C(=O)OC(C)(C)C)C1 C1(C(=O)NC2CCN(C(=O)Cc3cnns3)CC2CO)CCOCC12CCCC2 c1(CC(N2CC(CN=c3nc(SC)[nH]s3)C(C)C2)=O)nsc2ccccc12 C1(C(=O)NCCCN(C(c2n[nH]c(C)c2Cl)=O)CCO)COCC(C)(C)O1 c1(C(=O)NCC(CCNC(CN(C2CC2)CC)=O)O)ccc(C2CC2(Cl)Cl)cc1 Cc1cnc(C(=O)NCCC2(NC(C3CCC4CC4CC3)=O)CC2)cc1C CCC(CC)CC(=O)N1CCOCC(NC(=O)CCc2ccc(C)c(Cl)c2)C1 C(=O)(CCCCCC(C)(C)C)N(CCOCCNC(C(=Cc1cnc[nH]1)C)=O)C Cc1scnc1C(=O)N(CC(C)NC(=O)C(c1cn(C)nn1)N(C)C)CCO CCCCC(CCCC)C(=O)NCCOCCCNC(c1c[nH]c(=N)o1)=O CCC(C(=O)N1CC(NC(C)C)C1)NC(=O)C(C)=C1CC1 C1(CCNC(c2cnc(CC)s2)=O)CN(C(=O)CSCC(F)F)CC(C)O1 N1(C(=O)C=CBr)CC2CCN(C(c3ccc4ncnn4c3)=O)C2C1 N1(C(C2CC(SC)C2)=O)CC2(CCC(NC(=O)CC3CC(=O)NC(=O)C3)CC2)C1 CCC(F)(F)CC(=O)NC1CCCN(C(c2[nH]c(C)c(C)c2C)=O)CC1 N(C1CCCc2c[nH]nc21)C(C(CC1CCC1)NC(C(C(CC)CC)OC)=O)=O C1(CNC(C(c2cccnc2)NC(CSC(C)C)=O)=O)CCCC1C1CC1 CCC(C(=O)NC1(CNC(=O)CSc2nnc(S)s2)CC1)n1nccc1C Cc1cc(NC(=O)CC2(C)CCN2C(c2cc(CO)ccn2)=O)cnc1Cl C1(C(N2CC(NC(CC(=O)NCC#C)=O)C(C)C2)=O)CC12CCOC(C)C2 Cc1cc(Cl)cc(C)c1C(=O)NCCC1CN(C(=O)C(N2C(=O)CCC2=O)C)C1 c1(C(N2CC(CC(C)NC(=O)C(N3CCCCCC3)C)C2)=O)cccc(F)c1F C(=O)(CC(O)C(C)C)N(C1CCN(C(=O)CN(C(=O)C(C)C)C)CC1)CCCC Cc1nn(CC(F)F)cc1C(=O)NC1CCCC1CNC(=O)C(C)n1cncn1 N1(C(CC2(CNC(C(C)OC)=O)CC=CC2)=O)CCC(C)(CO)CC1 C(=O)(C1=C(Cl)CCOC1)NC(C(=O)NCC(C)OCC#C)c1ccco1 c1(C(=O)NC2C3CN(C(CC4(C(=O)OC)CC4)=O)CC32)cncc2c1CCCC2 c1(C(N(C2CCN(C(C3OCCN(C(C)C)C3)=O)CC2)C)=O)cc2sccc2s1 N1(C(C(N2CCCCCC2)C)=O)CCC(C)(CNC(=O)CCCc2cnn[nH]2)C1 CC(C)CC(C(=O)N1CC(O)CC1CNC(c1ccncc1)=O)N(C)C Cc1cc(N2CCC(NC(c3sc(CC4CC4)nc3C)=O)C(F)C2)nc(Cl)n1 Cc1cc(Br)cc(Cl)c1NC(=O)C(C)OC(c1ccc(N(C)C)cc1)=O C1(C(=O)OCC)CCN(c2nnc(C3CC3)n2CCCCOCC(C)C)CC1 c1(SC)cc(N2CCC(O)(C(C)NC(=O)Cc3cnccc3C)C2)nc(SC)n1 c1(C(=O)NCCC2CCC(NC(CSCCCC)=O)C2)ccc(O)nc1Cl C1(NC(c2c(C)c(-c3ccc(Cl)cc3)on2)=O)CCCCN(C(C2CCC2)=O)C1 N1(CC)CC(C(=O)NC2CCCC2NC(c2ccn(CC(F)F)n2)=O)NC1=O c1(C(N)=O)ccc(CC(=O)NCC2CCCN(C(C3CC(=O)N3)=O)C2)c(F)c1 C(=O)(C1=Cc2ccccc2C1O)NCC1(CNC(CC(CCCCC)C)=O)CC1 C1(C)(NC(C)=O)CCN(C(c2cccc(C)c2)C2CC2)CC1.n1(C)nccc1C c1(C(=O)NCC2C(NC(c3cc(OC)ncc3)=O)CCC2)cnc2nccn2c1 C1(NC(CCCOC)=O)CCCCCN(C(c2ccc(OC(F)F)cc2)=O)C1 N1(C(CCOC(COC)C)=O)CCCC(CN(CC(N2CCC(C)(C)C2)C)C)C1 c1(C(=O)NCCCCNC(C2(c3c(C)cno3)CC2)=O)cc2c(ccn2C)[nH]1 c1(C(=O)NC2(CO)CCCN(C(C3(C)CC(=C)C3)=O)C2)ccccc1N=[N+]=[N-] N1(C(c2c(OCC)cccc2)=O)CCC(NC(c2csc(C)c2)=O)C(O)C1 N1(C(C=C(CC)C)=O)CCCC(C)C1CNC(c1cc(C(F)F)nn1C)=O C1(NC(c2cc(C(F)F)ncn2)=O)C=CCN(C(C2(CO)CCOCC2)=O)C1 N#Cc1ccc(S(=O)(=O)N2CC3C(C2)N3C(c2cc3cccc(Br)c3[nH]2)=O)c(Cl)c1 c1(CC(=O)N(CC(CNC(c2c(C)snc2)=O)O)C)cnn2c1OCCC2 C(C(=O)N(CCNC(=O)C(F)n1ccnc1)C(C)C)(C(C)C)SC c1(COC)cccc(CC(=O)NCC2CCCN(C(c3c(C)ccn3C)=O)C2)c1 CC1COCC(C(=O)NC2CC(CNC(c3coc(Cl)c3)=O)C2)O1 c1(C(=O)NCC(CNC(c2c(CC)onc2C)=O)C)csc2nnsc12 C1(NC(=O)CN(C2CCC2)C(C23CCC(CO2)C3)=O)CCCCC1F c1(C(=O)NC2(COC)CN(C(c3cc(CC)c(C)s3)=O)C2)n[nH]c2c1CCSC2 c1(C(C)C)nsc(CC(N2CC(CC(C)(C)CNC(C3C(C)CC3C)=O)C2)=O)n1 C1(CNC(C=CCOCCOC)=O)CC2CCCC2N1C(=O)CC1CCC2CC2C1 C1(COC)(CNC(C2CC2CC(C(=O)C(O)(C2CC2)C2CC2)=O)=O)CCC1.C(C)(C)N c1(N2CCCC(NC(COC(CC)(C)C)=O)CC2)cnc(C#N)c(C#N)n1 N=c1ncc(C(=O)NCC(CNC(C23CCCC2(C(N)=O)C3)=O)CO)c[nH]1 C1(NC(CC=C=C)=O)CCCCN(C(c2ccc(NCCS(C)(=O)=O)s2)=O)C1 CCC(CNC(C1CC12CCC2)=O)(CC)NC(=O)Cc1nonc1C C1(NC(C(=O)NCC2CC2)=O)CC2(CCN(C(C3CC4CC4C3)=O)C2)C1 C1(CC)CN(C(C2CC=CC2)=O)CCC1CNC(=O)Cc1ccoc1 C1(CNC(c2cc(C)ncc2)=O)CC2CN(C(=O)C(C(C)C)OCC(C)C)CC12 c1(OCC(=O)NC(CNC(C2ON=C(C)C2)=O)(C)CO)cc(C)ccc1Cl N1(CC(c2cn[nH]c2)=O)CC2C(c3ccc(F)cc3)(C1)CS2(=O)=O S(=O)(=O)(c1ccc(Nc2cn(-c3ccccc3)nc2C)nc1)NCC(=C)C N1(C(C(=O)OCC)=O)CCC2(CC1)CC(NCc1c(Br)ccc(F)c1F)CCO2 CC1CN(C(C2CC2(C)C)=O)CCCN1C(=O)CCCc1c(F)cccc1F C1(CC=C)(NC(c2cncc(Cl)c2)=O)CCN(C(C2CCC(F)C2)=O)CC1 c1(C(N(C2CN(C(c3n[nH]c(C)c3C)=O)C2)C)=O)cnc2cccc(C)n12 N1(C(c2nc(CCC)oc2)=O)CCC(NC(=O)C(F)=C(C)C2CC2)C(C(C)C)C1 C1(C)(NC(C)=O)CCN(C(C2CCC2NC(c2ccnc(O)c2)=O)=O)C1 c1(C(=O)NCC(CN(C(c2cc(SC)oc2)=O)C)C)cc2c([nH]1)CCCC2 C(=O)(CC(C)C(F)(F)F)NC1CCC(CC(=O)NC(C)Cn2ccnc2)C1 c1(C(N2CC(O)(CNC(C(C)NC(C)=O)=O)C2)=O)ccc2c(c1)N(C)CC2 C1(C(C(=O)Nc2ccc(CC)cc2)N(c2ccc(C)cc2)C)OCCOC1(C)C C12(NC(C3CC(OC)C3)=O)CCC(C1)N(C(C1CCCC1OC(C)=O)=O)C2 C(C(C)C(C)C(=O)NCC(C)(C1CCC1)NC(=O)Cc1cncc(C)c1)OC Cc1csc(=O)n1CC(N1CC(N(C)C(C2(C)C=CCC2)=O)C(O)C1)=O C1(NC(CN(C(CCSCCC)=O)C2(C(=O)OC)CC2)=O)CC(C#N)C1 CN1CC2C(C(=O)NC3CCCC(CC(=O)NCCC4CC=CC4)C3)C2C1 Cc1nn(C)cc1CC(=O)NC1CC1CNC(=O)C(C)NC(=O)C(C)(C)C C(=O)(C(O)C(F)(F)F)N1CCC(C(C)(C)NC(C2CC(C(C)C)OCC2)=O)CC1 CC1(C(N2CC(CO)(NC(=O)CN3CC(C(F)(F)F)CCC3)C2)=O)CCCC1O n1(C(C)(C)C)cc(C#N)cc1NC(C1=CC=C(NS(=O)(=O)CC#N)C=CO1)=O Cc1nnc(O)c(C(N2CCC(NC(c3ccnnc3O)=O)C(C)(C)C2)=O)c1C C1(CNC(=O)C(O)C(F)F)CCCCN(C(=O)Cc2ccc(O)cc2)C1 Cc1c(F)cc(C(N2CCNCC2C(=O)Nc2c(F)cc(Cl)cc2Br)=O)cc1F C1(n2cc(C(CC)O)nn2)CN(C(C2CC=CCC2)=O)CC1.C1(C(N)=O)(N)CCC1 C1(C(N(C)CC2CCCN2C(C2(F)CCC2)=O)=O)CC(C)(C)CO1 N1(C(CCCOCC=C)=O)CCC2(COCCN2C(=O)Cc2cc[nH]n2)C1 N1(C(C=CCN(C)CC)=O)CC2CC1CN(C(c1c(Cl)sc(C)c1C)=O)C2 c1(C(N2CCCCC2CN(C)C)=O)cc(F)ccc1I.c12ccc(nc1)NC2 C1(C(N2CCC(CNC(c3cnc(C(C)C)o3)=O)CC2)=O)CC2CCC1NC2=O c1(NCc2ccc(C)c(F)c2)nc(=NCCC2CCCC2)[nH]c2c(C)nn(C)c12 C1(NC(CCNC(C)=O)=O)CC(NC(c2n[nH]cc2Br)=O)C12CCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CC(CC(=O)NCCN=S(C)(C)=O)C2(CC2)C1 c1(C(N2CC(N(C(CC(C)n3cccn3)=O)CCO)C2)=O)cn(C)c(C(F)F)n1 C(CNC(=O)CN1CCCCCC1)(CC(=O)N1CCCC(CC(C)C)C1)OC C=CCC(C(=O)NC(C)C(C)(C)CO)NC(=O)CCNC(=O)NC C1(NC(Cc2ccc(CC)cc2)=O)C2CC1CN(C(C1CC(=O)NC1(C)C)=O)C2 C1(C(=O)NCCC(=O)NCCN(C)CCO)CCCN(C(=O)N(C)C)C1 c1(C(=O)NCC23C(CN(C(C4(COC)COC4)=O)C2)C3)cccc2cccc(C)c12 c1(COC)ccc(C(=O)NC(C)C(CO)NC(=O)COc2cnc(Cl)cn2)cc1 Cc1cccc(C)c1C(O)C(=O)NCC(C)CNC(=O)CCSCC(C)C N1(C(C(C)n2cccn2)=O)CCC2(CC1)CC2CNC(C1CC2C=CC1C2)=O C1(C(=O)OCC=CC(=O)OC(C)(C)C)CC2(C1)CC1(CC(=O)C1)C2 c1(C(N2C(CC=C)(C(N3CC[SH](C)CC3)=O)CCC2)=O)ccc(C)cc1F c1(C(=O)NC(CC)(CNC(=O)CC2CCCCC2)CC)cc(F)c2[nH]nnc2c1 C1(CC(N2CC=CC(C(=O)NC3(CC4CCC4)CC3)C2)=O)CCC2CC2C1 C1(NC(C=CCCC(C)C)=O)CC2CC1N(C(=O)C(C)NC(N)=O)C2 c1(C(=O)NC2(CNC(c3c(C)scn3)=O)CCCCC2)ccc2c(c1)CCOC2 C1(C(N(CCOC)C)=O)CC1C1CN(C(c2coc(C(F)F)c2)=O)C1 C#CCC(C(=O)N1CCC(C(C)C)CC1)NC(=O)CC(C)c1ccco1 C(=O)(C(C)(C)n1ccc(C2CC2)n1)NCCCN(C(C1C(C)CC1)=O)CCO n1(CC(=O)NC(CNC(C(C2CCOCC2)C)=O)CO)ncc2ncccc12 CC(C)C(C)(O)C(=O)N1CC(NC(c2cnc(S)n2C)=O)C1 C(=O)(CCCCC=CC)NCCCN(CCCCCC)CC.C1(=O)C(C)N1 C#CCC(C)C(=O)NC(C)(C)CNC(=O)C(C)c1ccco1 N1(C(C2(C)C(C)CCC2)=O)CC2CC(NC(c3cc([N+](=O)[O-])nn3C)=O)CC2C1 C1(CNC(C=C)=O)CN(C(C2CCN(C)C(=O)C2)=O)CCC12CCC2 C12(C(=O)NC3(CC)CCOCC3)CCN(C(c3c[nH]c(C#N)c3)=O)CCC1C2 C1(NC(Cc2ccc(C)s2)=O)CC2(CCCN(C(c3ccnc(Cl)c3N)=O)C2)C1 n1(-c2ccn(CC)n2)nc(C(C)OC)nc1CCSC c1(C(N(C)CC2CCC2NC(=O)CC2CC=CC2)=O)ccn(C2CC2)n1 N1(C(CN(CCC)C)=O)CCC2(CC1)CC(NC(C1COC(C)C1)=O)CCO2 CCC(C)(C)CC(=O)N1CC2CCC1C2NC(c1ccc(F)c(C)c1)=O c1(C(=O)NC2(C)CCN(CCC(=C)C)C2)cc(C)nc(O)c1 c1(C(=O)NC2C(C(=O)OC)C2)ccc(C(F)(F)F)c(Cl)c1.c1(CN)ncccc1OC c1(CCC(=O)NC(CC=C)CNC(C2CCC3(CC3)C2)=O)csc2nc(C)cn12 N1(C(=O)NC2CCN(C(c3ccoc3)=O)C2)CC2(CCC1CO)CC2 N1(C(C2CCCN(C(C)C)C2)=O)CCC(O)(C(C)NC(C2CCCCC2)=O)CC1 C1(CNC(CCn2c(C(C)C)ncc2)=O)CC(C)CN(C(C2(C#N)CC2)=O)C1 C1(C(=O)NC2(CCCNC(C3CC(n4cnnc4)C3)=O)CC2)COC(=O)N1 C1(CNC(C2(C)CCC(C)C2)=O)CC2CCC(C1)N2C(C1CC(F)(F)C1)=O C12(NC(c3ccc(C(C)C)cn3)=O)CCC1CN(C(=O)Cc1c(Cl)cnn1C)C2 c1(C(N2CC(CNC(C(C)C)=O)C(C(F)(F)F)CC2)=O)ccc([N+](=O)[O-])cc1 N1(Cc2ccc(OCCC)cc2C)C(=O)CCN(CC2CCC(=O)N2)C1=O c1(C(N2C3CC(NC(c4cc(CC)no4)=O)C(C3)C2)=O)cc2cccc(O)c2[nH]1 Cc1cc(C(=O)NCC(C2CC2)N(C(=O)C(F)=CCCF)C)c(Cl)cc1Cl C(c1nc(C)c(C)[nH]1)=CC(=O)NCC(CC)NC(=O)Cc1ccc(Cl)nc1 c1(NC(c2c(NC(c3cc[nH]n3)=O)sc3c2CCC3)=O)cc(I)c(F)cc1F N1(C(CCCOCC)=O)CCN(C(N2CCN(C(=O)C(C)COC)CC2)=O)CC1 N1(C(C(C)=C(C)C)=O)CCCCCC1C(=O)NCC1CCCC1 c1(CCC(=O)NC2CC(CCC(=O)NCC(C#C)CC)C2)ccncc1OC C(CN=c1[nH]c(=NCC2(CSC)CC2)[nH]c2c1CC(C)CC2)=CCCOC c1(OC2(C(N3CCC(COC)CC3)=O)CCC2)nc(OC)nc(OC)n1 N1(C(CC2C(C(=O)OC)C2)=O)C2CCC1CC(NC(C1(C(C)C)COC1)=O)C2 c1(C(=O)NC(CNC(C2C(CC)OCC2)=O)(C)CC)ccc2c(c1)nc(C)n2C C(C(N=[N+]=[N-])C(=O)N1CCC(NC(C2(OC)CCC2)=O)C1)OCC c1(C(=O)NCC(CO)NC(Cc2c(C)nn(C)c2Cl)=O)cccc([N+](=O)[O-])c1 c1(OC)cc(C(=O)NC(C)C(CO)NC(C2CCC2C#N)=O)[nH]n1 N1(C(CN(CC)CC)=O)CCC(NC(c2cc(CO)cc(F)c2)=O)CC1C1CC1 C1(C(N2c3cnncc32)=O)CCC(C)(C)CC1.c1(NC(N)=O)cccc(N)c1.CO C1(NC(c2c(C(C)C)ccs2)=O)CCCC(NC(=O)CC(C)n2ccnc2)C1 CC1(C(=O)NC(CNC(c2csc(C(C)(C)C)n2)=O)C(C)(C)C)CC=CCC1 CCC(CC(=O)NCCCN(C)C(N)=O)C(C)(C)C.C1(=O)CC(C)N1 C1(CCNC(C2C(OC)CC2)=O)CN(C(=O)CNc2nccs2)CC(C)O1 Cn1cc(C(=O)NC2CCC2CNC(c2ccccc2F)=O)n2cncc2c1=O C1(CCN(C(c2c(C(C)C)ocn2)=O)C)CCCCN1C(=O)CCc1cscn1 C1(C2CCN(C(C3CN(C4COC4)C3)=O)CC2)(NC(c2cc(CO)[nH]n2)=O)CC1 N1(C(c2c(C)ncn2C)=O)CCN(C(=O)CN=S(C)(C)=O)C(C)C1 N1(C(CN2CCN(C)CC2)=O)CCC(F)(C(=O)NCCc2cnccn2)CC1 C(C(CC(C)C)C(=O)NC1CCCC1(C)CO)NC(c1c(CC)n(C)cc1)=O c1(CNC(Cc2ncc(-c3ccc(=N)[nH]c3)cn2)=O)cccc2c1OCC2 CC1CCC(CNC(c2sc(F)cc2Cl)=O)CN1C(=O)CNC=O c1(C(=O)NCC2C(NC(C3(CC=C)CCCC3)=O)CCC2)cnn(C)c(=O)c1 Cc1ccc(C(N2CC(NC(=O)C(c3cccnc3)C)CC2C)=O)cc1Cl N1(C(c2c(CC)cno2)=O)C2CCC1C(NC(C1CCCC1)=O)C2 N1(C(C2CCc3cn2nn3)=O)CCCOC(COC)C1.c1(CC)cc(NC)nn1C C(C)(CN=c1[nH]c(Cl)nc(N2CCOCC2)c1C)Oc1ccc(C)cc1C c1(C(C)Nc2cc(N3CCCC(C(N)=O)C3)ncn2)nc(Br)sc1C Cc1cc(=NCC2CN(C(=O)CCc3cc[nH]n3)C2)nc(O)n1-c1ccccc1 C1(NC(C2(CC(C)=O)CC2)=O)C2CCC(C2)C1C(=O)NC(c1ccccc1)C#N N1(c2snc(C)c2C#N)CC23CCCC2(CN(C(=O)C(O)CC(C)(C)C)C3)C1 C(=O)(CCC(C)(C)C#N)N1CCCCC(CNC(CC2ON=C(C)C2)=O)C1 C1(C(=O)N(C)CC2CCN(C(c3cccc(N)c3)=O)C2)(OCC)CCOCC1 c1(NC(c2ccc(C3COc4ccccc4O3)o2)=O)nc2cc(Cl)ccn2n1 C(CC(C(F)F)N(C)C)N(C)CCc1ccc(F)cc1.C(CF)N c1(NC(=O)NC(C)(CCCO)c2nnnn2CC(F)F)ccccc1CN(C)C CC(CC(=O)NC1CCN(CCCNC(=O)C=CC2(C)CCOCC2)C1)C(F)(F)F C(CC(=O)NCCc1ccnc(O)c1)(C(F)(F)F)NC(C1CC(=C)C1)=O c1(CNC(c2n(CCCCCC)nnn2)(C2CCCO2)C)cc(C)ccc1Cl C1(C(N2CCN(C(C3CCN(C(CC)=O)CC3)=O)CC2)=O)CCCC2C1C2(F)F N1(C(c2cncc(COC)c2)=O)CCN(C(C2(OC)CCCCC2)=O)CC1CF N1(C(CCc2cnc(C)o2)=O)CCC(C(=O)NC2CC2c2cncs2)C(C)(C)C1 CC(C)(CC(=O)OCc1cnco1)C1CCCCC1 C=C(C)CC(C(=O)NCCN1CCCCC1)NC(=O)CCOCC(=O)OC CC1CN(C(c2cncc(CO)c2)=O)CCC1N(C)C(c1ccc(=N)[nH]c1Cl)=O C1(N(C(c2sc(CCC)c(CC)c2)=O)C)CCN(C(c2cc[nH]n2)=O)CC1C c1(C(=O)NCC2N(c3nnc(C)s3)CCC2)cc(F)c(F)cc1F S(=O)(=O)(CC(=O)NC12CC(NC(c3cncs3)=O)(C1)C2)N(C)C C=C(C)CC(C(=O)NCCCOCC(=O)NCC(C)(C)SC)OC C1(F)(CNC(c2ncccc2Cl)=O)COCCN(C(c2cn(CCF)nn2)=O)C1 C1(C)(CNC(c2c(C(C)C)ocn2)=O)CN(C(=O)CN(C2CCSC2)C)CCO1 C1(NC(C2(CC=C)CCC2)=O)CC(O)CN(C(c2c[nH]nc2CC2CCC2)=O)C1 CN1CCN(C(c2ccncn2)=O)C(CNC(C2CC23CCCC3)=O)C1 N1(C(C2(N(C)C)CCCCC2)=O)CC(NC(=O)CCC2CC2(F)F)C(C2CC2)C1 C1(CC(=O)NCCC(=C)C)C2CCCC2N1C(=O)CC12CCCC1C2 N1C2CCC1CN(C(=O)CN(C)CC)CC2.CCC(CC)CCC=O Cc1c(C(=O)NC(C2CCOC2)CNC(c2ccoc2C2CC2)=O)cncc1F N1(c2cc(N(C)Cc3ncc(Br)cn3)nc(C(C)C)n2)CCC2CN(C)CC2C1 N1(C(c2c(SCC)cncc2)=O)CCC(NC(c2ccon2)=O)C(F)C1 C1(F)(NC(=O)OC(C)(C)C)CC(C(=O)NC2(NCc3ccsn3)CCOC2)C1 c12ccc-1cc2.C(=O)(C(C)CF)NC(C(C)N)C.C(=O)CSC(F)F Cc1nn(C)cc1C(=O)NCC1CN(C(=O)CNC(c2cscn2)=O)CC1C c1(C(N2CCNC(=O)C2CCO)C(=O)NCCC)cccc2nc(C3CC3)[nH]c12 N1(C(c2cnc(OCC)nc2)=O)CC2CC1CCC2NC(=O)C(C)SC c1(C(=O)NCCC(C)N(C(CCN(CC)CC)=O)CCO)ccc(OC)nc1 N1(C(CNC(CC(C)OC)=O)=O)CCCC(C)(O)C1 C(=O)(CCCCC(C)C)NCC(CC(F)(F)F)NC(C(c1c(C)noc1C)C)=O C1(C(N2CCC(CCNC(c3nnc(O)cc3O)=O)C2)=O)Cc2ccccc2S1 n1(CC)cc(CC(=O)NCCC2CCC(NC(=O)CNCC=C(C)C)C2)cn1 C(CC(C)C(=O)N1CCN(C(C2CC(C)CCO2)=O)CC1)OC C1(C)(CNC(c2c(OC)nsc2)=O)CN(C(c2scnc2C(C)(C)C)=O)CCO1 c1(C(N(C(C(C)Oc2cc(Cl)cc(Cl)c2)=O)C)C)nc2ccccc2s1 C1(CNC(CC2(CNC(CC3CCN(C)C3)=O)CC2)=O)CC2(CC2)CO1 C1(CNC(c2cc(C)nn2C)=O)CCC(C)(C)CN1C(=O)C(O)CC(N)=O c1(C(=O)NCC(CC2CN(C(COCC#C)=O)C2)(C)C)cc2ccc(Cl)cc2o1 c1(NC(n2cnc3sccc3c2=O)=O)ccc(S(=O)(=O)NC2CS(=O)(=O)C2)cc1 Cc1cc(F)sc1C(N1CC(CNC(=O)CNC(c2cccc(O)c2)=O)C(C)C1)=O N1(C(C2(CC)COC2)=O)CCCC(C(N2CCN(CCF)CC2)=O)CC1 C1(C(=O)OC)(NCc2cn(C)nc2OCCF)CCC12CCC2 c1(OC)cnc(C(=O)N(CCCNC(c2cccc(Cl)c2Cl)=O)C)c(F)c1 N1(C(C2CC(CC)C2)C(=O)NC(C)CC)CCOC(c2n[nH]c(C)n2)C1 C12(C(=O)NC3(C)CN(C(=O)CC4CCCOCC4)C3)CCCC1C2Br c1(NC2CCCN(CC)C2)nc(C)cc(=NCC2(CC(N)=O)CCCC2)[nH]1 N1(C(C(CC)CC)=O)CCC(N(C)C(c2cnc3ccccc3n2)=O)C2(CC2)C1 c1(C(=O)NCC(CN(C(C2(OCC)CCC2)=O)C)O)cnc(OC)cc1OC N1(CC(C)C)CCN(C(c2conc2CNC(=O)CC2CCCCO2)=O)C(C)C1 c1(C(N2CC(NC(C3(C=C)CCC3)=O)C(F)CC2)=O)cc2c(F)cc(C)cc2[nH]1 c1nc(NCc2ccns2)cc(C2(C3CCCCO3)CCC2)n1 c1(NC)cc(C(=O)NCC2=CCN(C(=O)CCCNS(C)(=O)=O)CC2)ccc1F CCC(CC(=O)N(CC(C)(C)NC(=O)CCC(F)F)C)CC(F)(F)F c1(C(N2CCC(NC(Cc3n(C(C)C)cnn3)=O)C2C)=O)cc2occc2n1C C1(C(N(C2CC3(CC3)C2)C)=O)CCN(C(=O)c2cnnc(O)c2)O1 C1(CNC(c2n(CCC)ncc2)=O)CC(C)CN(C(c2ccc(=N)[nH]c2C)=O)C1 CC1(C)C2CCC(C(=O)NC3CC3CNC(c3cnc(O)c(F)c3)=O)C1C2 c12cccc(c1)S(=O)(=O)N2.C1(C(=O)Nc2cc(CC)no2)CC2(C1)CC(CO)C2 C1(NC(=O)CC2CC2)CC2CCC1(NC(=O)Cc1ccc(Cl)cc1)C2 C(=O)(C1=NOC(C)(C)C1)NC(CN(C(c1c(C)nc(-c2cnccn2)s1)=O)C)C O(NC(=O)C(Cc1ccccc1Br)NC(=O)CC1C=CCCC1)CC=C(C)C n1(CC(=O)NC(CN(C(C2C(OCC)C2C)=O)C)C)cc[n+](C)c1 c1(CC(CN(C(=O)Cc2cncn2C)C)NC(C2CC2C(C)(F)F)=O)ccccc1 CCCC(C)(CC)C(=O)N1C2CCC1CC(CNC(c1cc(Cl)ncc1O)=O)C2 c1(CC)cnccc1C(=O)N(C1(CC(=O)N(C)CC)CC1)C C1(C(C)NC(C(CC)n2cncn2)=O)(C(=O)NC23CC(C2)C3)CCOCC1 N1(C(C=CCC)=O)CC2CCC(NC(c3coc(C(F)F)c3)=O)CC2C1 c1(C(=O)NCC2(NC(c3cncc(OC(C)C)c3)=O)CC2)ccc2nsnc2c1 C(C1CCCC1)=CC(=O)NCCN(C(c1cn[nH]c1)=O)C1CC1 Cc1ccsc1CC(=O)N(CC(C)NC(=O)C(n1nnnc1C)C1CC1(Cl)Cl)C N1(C(C2CC(OC)C2)=O)CCC(N(C)C(c2cnc(C)[nH]2)=O)C1 C1(CCOC)(NC(=O)C(C)CCc2cccc(F)c2)CCN(C(=O)C(C)CO)C1 c1(C(=O)NCCOCCN(C)C(c2cc(C(F)F)no2)=O)ccc(O)c([N+](=O)[O-])c1 CCS(=O)(=O)c1cccc(NC(=O)NCCOCCO)c1 N1(C(C=CCN(C)CC)=O)CC2CCOC2(CNC(=O)Cc2cnccc2C)C1 C1(CNC(c2ccc(CNC(Cc3c(C)ncs3)=O)o2)=O)CCOC(C)C1 c12cccc(Cl)c1NC2=O.c1(COC)ccc(CO)[nH]1.C12CC1C(=O)N2 C1(C(=O)NC(CO)C(=O)NCC2CCOC2)C2CCCC12 C1(=O)CCC(C)CNC2(C(=O)OC)CCN1C2.C1(c2cnn(C)c2)C2CCCC12 C1(CC(=O)NCC(C)(C)CNC(=O)CCOC2CC2)CCC(=O)NC1 Cc1cccc2c(C(=O)N(CC(C)(C)CNC(=O)C(C)(C)C(C)C)C)c[nH]c12 C1(N(C(C2C(OC)CCCC2)=O)C)CCCCN(C(=O)COc2cn[nH]c2)C1 c1(OCC(N2CCC(CNC(CCC=CC)=O)CC2)=O)cccc2ccccc12 C(=O)(C(C)(C)C(C)(C)O)N1CCCCC(NC(c2c(F)ccc(C)c2)=O)C1 Cc1cc(C)c(C(=O)NC2(CNC(C3CCC(C)CC3)=O)CCCCCC2)cn1 N1(C(c2c(OC)nsc2)C(=O)NC(C)(C)C)CCC(Cc2nnc(C)s2)CC1 c1(OCC)cccnc1C(=O)NC(CNC(=O)Cc1ccc(Br)cn1)CO C(=O)(C#CC1(C)CCCO1)N1CCC(C(C)C(N2CCC(CO)C(C)C2)=O)CC1 c1(C(=O)NCc2ccc(NC)cc2)cccc2c1OCCN2 N1(C(C(CCO)N(C)C)=O)CCC2(CC1)CN(C(=O)CC1=CCCC1)CCO2 C1(C)(C(N2CCN(C(C(C)(C)C)=O)CC2)=O)CC2CCC1O2 C(=O)(C(O)CC(C)C)NC1CC(F)(CNC(CCC=C=C)=O)C1 N1(C(C(C)OCCCC)=O)CC2C(CN(C)C(c3ccc(CN(C)C)[nH]3)=O)C2C1 c1(C(=O)OCC)ccsc1COC1CCCC1NC(C1OCCC1CC)=O C(=O)(C(C)(C)CCC#N)NC1C(C(F)(F)F)CCN(C(CC(CC)OC)=O)C1 c1(-c2cc(C)c(F)c(C)c2)ncn2c1CN(C(=O)C(C)(C)C)CC2 CC1C(C(N2CCN(C(=O)CS(C)(=O)=O)CC23CCC3)=O)OC2CCCCC12 Cc1ccc(CC(=O)NCC2CC2NC(=O)Cc2cc(O)nc(O)n2)cc1C c1(OC)cccc(NS(=O)(=O)CC2CC2C(=O)OC(=O)C2CC2)c1 c1(NC(=O)NC)ccc(C(=O)NC(C)C(C)NC(c2cc(C#N)no2)=O)nc1 CCCCCC(F)C(=O)NC(CCCC)C(=O)N1CCC1COC N1(C(C(C(C)O)C)=O)CCC2(CCN(C(=O)C=Cc3ncc[nH]3)CC2)C1 C1(CCC)CCCC1C(=O)NCC12CC(NC(c3cn(C4CCOC4)cn3)=O)(C1)C2 N1(C(C(C2CCCC2)OCC)=O)CCN(C(c2cccnc2CC2CC2)=O)CC1 c1(OC)ccc(Cl)c(C(N2CC(NC(=O)C3=CCCS3)CCC2C)=O)n1 Cc1cc(C=CC(=O)NC2CCN(C(=O)CC3CC(F)(F)C3)CC2)on1 C1(C)(CNC(C2CCC(CC)O2)=O)CN(Cc2cccc(C)c2Cl)CCO1 C(=O)(C(C)S(C)(=O)=O)NCC(C1CCCC1)NC(Cc1c(C)n(C)cn1)=O C(=O)(CC1=CCOCC1)N1CCC(CNC(C(C)OCCCC)=O)C1 CCC(CC)CCC(=O)N1CCC2CC2(C(=O)NCc2cnn(C)c2C)CC1 c1(CC(=O)N(C)CCC2CCN(C(=O)CNC=O)CC2)cc(Cl)c2c(c1)OCCO2 C1(CC(=O)NCCC2CCC(NC(c3cncc(CO)c3)=O)C2)CC2(CC2)CO1 C1(C(=O)NCC(C(CC)C)C)CN(C)CCN1C(=O)CN(C)C N1(C(CC2CCC(OC)CC2)=O)CCCCC(CNC(C2CCS(=O)(=O)C2)=O)C1 C(C(C)N=c1cc(C#N)nc(C)[nH]1)NC(C1(OC)CCC1)=O C(=O)(C1=NNC(=O)CC1)NCCC1N(C(CC2N(CC)CCOC2)=O)CCOC1 c1(C(N2C(C(N(CC(O)CO)C(C)C)=O)CC(O)C2)=O)cc(F)cc(Br)c1 C1(NC(CN=[N+]=[N-])=O)CC=CCC1C(=O)NCCCOC(=N)O c1(CNC(=O)OC(C)(C)C)cc2c(C#N)cccc2[nH]1.CON1CC(C=O)CC1=O C1(C(=O)NC(c2nc(-c3ccccc3Br)no2)C)C2CNC(=O)C12 c1(OC)ccc(OC)c(CC(=O)N(C)CCOCCNC(=O)CC2CC(C)C2)c1 C1(c2ccccc2F)(NC(=O)NC2CC(CC)(CC)C2)CCCCC1 CC(C)CC(CNC(c1cnc(-c2ccsc2)s1)=O)NC(=O)COCC(C)(C)C N1(C(C2C(COC)C2)=O)CC2CN(C(C3(OC)CCC(C)(C)CC3)=O)CC2C1 C(=O)(CCN(OC)C(=O)C1CC(NC(=O)CC2CCC(=O)N2)C1)OC(C)=O C1(CC(=O)NCC(C)CN(C)C(c2ccnc(NCCO)c2)=O)NC(=O)NC1=O Cc1cnnc(O)c1C(N1CC(C(O)C(=O)NCC2OC3CCC2C3)C1)=O C#CC1CN(C(=O)CCC(C)(C)F)CCN1C(=O)C(C)C(=O)c1cccc(OC)c1 C1(CN(C(c2cnn(C)c2)=O)CC)CCCN1C(=O)CC1CCSCC1 C1(COC)CCCCCN1C(c1ccc(-c2ccc(C)c(N)c2)cc1)=O C1(CNC(=O)CNC(c2cscn2)=O)CCCCN1C(=O)C=C(C1CC1)C1CC1 CN1CC(=O)N(CC(=O)N(CCNC(C2CCCC2O)=O)C2CC2)C1=O C1(C(N(C2CCN(c3nnc(O)s3)C2)C)=O)CC(c2ccccc2)=NO1 O(NC(=O)C1=NOC(CNC(c2cscc2C)=O)C1)CC(=O)OC c1(CNC(C2C(F)(F)C23CC3)=O)ccc(C(N2CCCC2(CO)CO)=O)cn1 N1(C(C=C)=O)CC(NC(=O)C(c2ccccc2)F)C(C)C1 c1(CC)nc(O)c(C(=O)NC2CCC(CNC(C3(CC4CC4)CC3)=O)C2)cc1C N1(C(C2CCCC(OC)C2)=O)CCN(C(=O)C(CC(C)C)NC(N)=O)C2(CC2)C1 C(C(CC(F)(F)F)NC(C1CC(=O)NC(C)C1)=O)NC(C1(SC)CC1)=O C(C)(CCN=c1nc(C(F)(F)F)[nH]s1)NC(c1c(C)ccc(C)c1)=O C1(c2oc3ccc(C)cc3n2)NC(=S)N(CCCO)C2=C1C(=O)OC2 C1(CCNC(C(C)N(C)C(=O)Nc2cc[nH]n2)=O)CCCCC1 c1(CC#N)ccc(C(N2CCC(NC(CS)=O)CC2)=O)cc1.C1CCCS1 C1(C=O)CCC(C)(C)CO1.[nH]1cc(CN(C)C(=O)O)nn1.O(C(=N)O)CCCOCCOC CN=c1nc(N(CC(=O)NCC(C)C)C)[nH]c(=NCCS(C)(=O)=O)[nH]1 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCC(N(C(CCCC=C)=O)CCC)C1 CC(C)CC(C(=O)NCC(O)CNC(c1cn(C2CC2)cn1)=O)C(C)C N1(CC)N=C(C(=O)NC2CCC2NC(c2cscc2C(N)=O)=O)CCC1=O c1(C(=O)OCC)c(F)c(NC(C2CN(S(=O)(=O)N(C)C)C2)=O)cc(C)c1Br c1(N2C(C3(C)CC3)CCC2)nc(NC(C2CCCCS2(=O)=O)=O)nc(=N)[nH]1 Cc1[nH]nc(C(N2CCOCC2CNC(=O)CCCN(C)C(C)C)=O)c1N N1(C(c2cn(C=C)nc2)C(=O)NC2CCC2)CCN(C)C(=O)C1CCO S(=O)(=O)(c1cnccc1N1CCCC(CC(N)=O)C1)NCC(C1CCCC1)OC C(=O)(C(CC1CCC1)NC(CSCCOC)=O)N(C(=O)C(C)C)CC1CCC1 c1(NC(c2ccc(-n3cnnn3)cc2)=O)cccc(Cl)c1CO C1(NC(c2cnn(C)n2)=O)CC2CC(C1)N(C(=O)CNC(c1ccco1)=O)C2 C1(C(=O)NC(CNC(c2ccc(-c3cccs3)[nH]2)=O)C2CC2)CC2CC2C1 C(=O)(C1=CCCN(C(=O)CC2CCC(=O)CC2)C1)Nc1c(N(C)C)nccc1 c1(CNC(CC(=O)N)=O)cc(C(=O)OCC)cs1.C1CC(N2CCCC2)C1.OC c1(C(=O)NCC2C3N(C(C(C)CF)=O)CC(CC3)C2)cc2cccc(F)c2o1 c1(C(=O)NC2CN(C(C=CCOC)=O)CC2C2CC2)cc2cccc(F)c2o1 c1(N2C(C)CC(CNC(c3c(C)nn(C)c3)=O)C2)ccc([N+](=O)[O-])cc1Br C12(CCNC(Cn3c(C)nnn3)=O)CCC(C1)N(C(=O)C1=COCCC1)C2 Cc1ncc(C(=O)NCC(=O)NCC2(CO)CCOC2)c(C)n1 C1(C(N2CCN(C(CC(CC)OC)=O)CC2CC)=O)CCn2c(O)nnc2C1 N1(C(c2ccc(=NCC)[nH]c2)=O)CC2(CCN(C(=O)OC(C)(C)C)CC2)C1 C12(C(N3CCCC(N(C)C(c4ccncc4F)=O)C3)=O)C3C4C1C1C2C3C41C#N C1(NC(CC(C2CC2)NC(CC(C)CN(C)C)=O)=O)CNC(=O)C1(C)C C12(NC(c3c(C(C)C)sc(Cl)n3)=O)CCCN(C(=O)CSC3CC3)CC1C2 c1(CCC(=O)NCCOCCCNC(=O)Cn2cncn2)ccc2c(c1)CCO2 Cc1nc(NCCN2CCOCC2C)cc(N2CCCC(C#N)C2)n1 CC1CCN(C(=O)CCS(C)(=O)=O)C(C)C1NC(c1cccc(Cl)c1)=O c1(C(=O)NCCOCCNC(CC2CC(OC)C2)=O)ccc(Cl)c2ccccc12 C1(CC=C)(NC(=O)CN2CC3CC3C2)CCN(C(C2(CSC)CCCCO2)=O)C1 C1(C(F)(F)F)(NC(c2cn(C3CCNC3)nn2)=O)CCNCC1 c1(OC)ccc(C(=O)NC2CCCN(C(c3csc([N+](=O)[O-])c3)=O)C2C)cc1F C1(NC(c2c(OC)ncc(F)c2)=O)CN(C(=O)COC(F)F)CC12CCOCC2 c1(C(N(CCNC(C2N(C(C)=O)CCC2)=O)CC)=O)ccc(C)c2c1NCCC2 N1(C(CC(C)C2CC2)=O)CCCC(C2CC2NC(=O)COC(F)F)C1 c1(C(=O)NCCCC)ccc(NC(C2CCCN2C(c2cccn2C)=O)=O)cc1 Cc1n[nH]c(C)c1C(=O)NC1CCC(N(C(=O)CC2CCCCC2C)C)CC1 N1(C(c2c(SC)scc2)=O)CCC(N(C)C(c2ccc(C)o2)=O)CC1 c1(C(=O)NCCOC2CN(C(C(C)CC(N)=O)=O)C2)cnn2cc[nH]c(=O)c12 c1(C(n2cc(CC3(O)CCOC3)nn2)CNC)ccccc1 c1(C(=O)NCC2C(NC(CNC(CCCCC)=O)=O)CC2)cc(O)nc(C)n1 N1(CC(=O)NCCOC)CCN(C(C2OCCC2C)=O)CC1 Cc1ncc(CCNC(N2CCC(OCc3cn(C(C)C)nn3)C2)=O)[nH]1 C1(C(=O)NC2(CNC(C(C)CC3CCCC3)=O)CCCC2)CC2CC1CC2(F)F c1(NC(=O)NC(CCCC)c2cccnc2)ccc(N2CCCCCC2)nc1 C1(C(N2C(CNC(C3CCC34CCC4)=O)CCC2)=O)CC2CCC(C1)S2 c1(SC)ccc(C(N2CC(F)(CNC(=O)CCN3CCCCC3=O)C2)=O)cn1 CN1CCCC1C=CC(=O)NC(C1(O)CCCCC1)C(=O)NCCN1CCCC1 C(=O)(C(C)C(C)NC(C1CC2CC2C1)=O)NC(c1ccccc1Br)C c1(NCc2cc(C)ncn2)nc(N(C)CC2CN(C)C2)c2c(ncn2C)n1 C=CC(F)(F)C(=O)N1CCN(CC(C)NC(=O)C(c2ccc(F)cc2)F)CC1 c1(-n2c(C(c3ccn(C)n3)NCC(CO)OC3CCCC3)nnn2)ccc(F)cc1 c1(C(N(CCCNC(=O)C(F)CC2CCOC2)CC)=O)cnc(C(F)F)c(F)c1 c1(NC(C2N(C(CCCC(C)C)=O)CC(O)C2)=O)cccc2occc12 N1(C(C2C(=C)C2)=O)CC2CCC1CN2C(=O)CN(C)C(C)C C(=O)(C(C)(F)C(=O)NCCOCCO)NCCN(C(=O)CC(C)CCC)CC C1(C(=O)NC(CN(C(=O)COCCCOC)CC)C)CCc2ncnn2C1 C1(C(=O)NCC(C)N(C(c2n(CC)ncc2)=O)C)CC=CCC1C(F)(F)F N1(C(C(c2cc(C)sc2)(C)C)=O)CC2CC(NC(C34CC(C)(CO3)C4)=O)CC1C2 CCC(C)CCN=c1[nH]c(N(CC(N)=O)C)nc2c1CCCCCC2 C1(O)(C(=O)NC(CC)CNC(=O)C(C#N)C2CC2)CCCC(C)(C)C1 N1(C(CC2(OC)CCC2)=O)CCC2CN(C(c3nocc3Cl)=O)CCC2C1 N1(C(c2c(C)oc(C(C)C)n2)=O)CCCC12CCN(C(=O)C(C)CF)C2 C(=O)(C1=CS(=O)CCC1)NC1(CN(C(CCc2nnc(C)n2C)=O)C)CC1 C(=O)(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(C)C)N(CCSC)CC C1(CNC(c2cc(CNC(C3(C(=O)OC)CC3)=O)[nH]n2)=O)CCCCC1C c1(OC)ccc(S(=O)(=O)N2CCOCC(NC(c3cc(F)cc(I)c3)=O)C2)cn1 C(C(CN=c1ccnc(C2CCC2)[nH]1)C(F)(F)F)NC(C1(COC)CCCO1)=O C12(C(N(CC(C)NC(c3cnn(C)c3C(F)(F)F)=O)C)=O)CCCCC1C2(F)F N1(C(c2cc(CC)n(CCO)n2)=O)CC2CCC1C1CN(C(=O)C(F)CC)CC21 C(=O)(CS(=O)(=O)CC)N1C(CNC(=O)C(C)NC(N)=O)CC(OC)C1 C1(C(N2C(CN(C(=O)CS(=O)(=O)N(C)C)C)CCC2)=O)CN2CCN1CC2C CCC(C(=O)N(C(C(=O)NCCCC(=O)NC1CC1)C1CC1)C)N1CCCC1=O CCCC(C(=O)N1CC=CC(NC(C2CCC3CC23)=O)C1)c1ccccc1 C(=O)(CCCC(F)(F)F)N1CC(O)(CCNC(C(c2ccc(O)cc2)(C)C)=O)C1 CN1CCCC(C(N2CCC(C(O)CNC(C3(CO)CC3)=O)CC2)=O)C1 C1(C(N2CCC(CCCO)C2)=O)(COC)C=CCN1C(c1sc(O)nc1C)=O CCCCCCCCCCCCNC(c1nnnn1CC(F)F)c1ncco1 C(C(=O)N1OC2C=CC1CC2)=CCC1N(C(c2c(C)con2)=O)CCC1 C1(NC(c2c(SC)cn(C)n2)=O)CC12CCN(C(c1ccns1)=O)CC2 C(CC(C(=O)N1CCC1CN(C)C)NC(c1cnc(NC)s1)=O)=CC C(=O)(CS(=O)(=O)CC(=O)N(CCCNC(=O)CC1CC2(CC2)C1)C(C)C)OC C1(CC(=O)NCCCCN(C)C(C2CC3(CCC3)CO2)=O)CCCCC1(F)F N1(C(COCC(C)C)=O)CC2(CCCC2)C1C(=O)NCCOC(F)F CCC(C)CCCC(=O)NCC12CC(CN1C(c1cc(C)c(N)cc1F)=O)C2 c1(OC)cc(-c2ncccc2NC(c2cc(-c3ccccc3)no2)=O)cc(C)c1 C1(NC(CCC(C)C)=O)CC12CCN(C(c1cc(C)c(C(F)(F)F)s1)=O)C2 NS(=O)(=O)c1ccc(C(N2CC=CC(NC(c3cncn3C3CC3)=O)C2)=O)cc1 C(=O)(C(C)CCC(C)(C)C)N1CC(CC=C)(NC(=O)C2=C(C)CC2)C1 N1(C(C2(OC)CCC2)=O)CCC2(CCCN(C(c3cnncc3C)=O)C2)C1 c1(C(=O)NC(C(=O)OC)C2(O)CCC2)cscc1C(=O)OC(C)(C)C C1(NC(Cc2scc(C)n2)=O)CCCCN(C(=O)CCOCC(F)(F)F)C1 C12(CNC(C3CC(C)(O)C3)=O)CCC1CN(C(c1cccc(F)c1Br)=O)C2 CCS(=O)CC(=O)N(CCCO)OC.C1C(C)CCN1C C(=O)(C1=CC2C=CC(C1)C2)NCC1(O)CCCN(C(c2n(C)nc(CO)c2)=O)C1 c1(C(=O)NC2CCCN(Cc3c(OC)cccc3O)CC2)cccn2ccnc12 c1(NC(C)CCn2cncn2)nccc(=NCCc2cccnc2Cl)[nH]1 c1(C(=O)NC2(CNC(C3CCC(C)S3)=O)CCC2)cc2cccc(Cl)c2o1 CCC1CCN(C(=O)OCC2CC(=O)N(C(C)C)C2)c2ccccc21 c1(CC)ccc(C(N2CCC(CN(C)C(c3ccc(N)c(O)c3)=O)C2)=O)cc1F C(CCC(O)C(=O)NC1CC1C1CCC1)NC(Cc1c(C)n[nH]c1C)=O Cc1ccnc(C(C)(C)C(=O)NCC(F)CNC(=O)C(C)NC(=O)OC(C)(C)C)c1 c1(N2CCC(CCC)C2)nc(=NCCCCCOC)[nH]c2c1CSC2 C1(C(=O)NCCC(C(C)C)NC(C(CCC)C)=O)CCn2cncc2C1 C12(CNC(=O)Nc3ncccc3OC3CCOC3)CCCN(CC1)C2 c1(N2CC(C(C)N(C3(C)CCCO3)C(=O)CSC(F)F)C2)ccncc1C#N C(=O)(C(C)CS(C)(=O)=O)NC1CCC(N(C(c2cc(C#C)nnc2)=O)C)CC1 Cc1ncc(C(=O)NCCC2(O)CN(C(=O)CC3CCCC(C)C3)C2)c(C)n1 C(=O)(CCCCCOC)NCCC(=C)CNC(c1ccc(N2CCCC2)cc1)=O C1(CNC(c2c(CC)c(C)ccc2)=O)CCN(C(c2nc(Cl)oc2C)=O)CC1C CN1CCN(C(C2COCCN(CC3(C)CCCCC3)C2)=O)CC1=O C(=O)(C(CC)C(C)(C)CC)N1CC(C=C)C(NC(c2cc(C)nc(C)n2)=O)C1 c1(CC(=O)N)c(Cl)cncc1Cl.c1(C(=O)OC)cc(C(=O)NC2CC2N)cs1 c1(CC)ccc(C(N2CCC(NC(=O)CC(C)C)C(CC)C2)=O)cc1F N1(C(CCOCC#C)=O)CC2CCC(Nc3ncnc4sc(C)nc34)C2C1 C1(C(=O)NCc2oc(C(=O)NCC(CCC)CO)c(C)n2)CC(=O)C12CCC2 Cc1nc2ccccc2nc1C(=O)NC1CN(C(c2ccccn2)=O)CC1O C1(CCC)(C(=O)OCC)CCN(C(=O)Cc2ccncc2C)CC1.n12cc(nn1)C2 Cc1cc(CCCC(=O)NCC2(NC(=O)CCc3ncccn3)CC2)c(C)s1 C1(NC(C=CC(N)=O)=O)CCN(C(=O)C=Cc2ccc[nH]2)CC12CCC2 Cc1ccc(C(=O)NCC2CCCN2C(=O)Cc2nn(C)cc2Br)cc1N CC1=C(C(=O)N2CCOCC2CNC(c2ccc(C(F)F)cc2Cl)=O)CCCC1 C#Cc1cccc(CC(=O)NC(Cc2ccccc2)CCNC(=O)CN(C)C)c1 c1(CC)cnc(C(=O)NC2CCC(NC(=O)C(c3ccccc3OC)C)C2)cn1 C(C(C)(C)CNC(C1CC1(c1ccccc1)F)=O)N(C(CNC(=O)OC)=O)C c1(NCCNC(=O)Nc2ccc(C#N)nc2)ccc2oc(O)nc2c1 C(C)(CCC(=O)NC(c1cnn(C)c1)C(=O)NC1CC(=C2CC2)C1)OCC N1(C(C(=O)NCc2cc(C)sc2Cl)=O)CCNC(=O)C1c1cccs1 C(=O)(CCCCC(C)(C)OC)NCC(C1CCC1)NC(C1(CC)CCCCC1)=O c1(C(=O)N(CC(N2CCCC(N(C)C)CC2)=O)C2CC2)cc(Cl)ncc1F CCC(CC(=O)NC1CC(OCC(N2CCN(C)CC(O)C2)=O)C1)C(F)F N1(C(c2cn(CCOCC)nn2)=O)CC(NC(=O)C=CC(C)CC)C(O)C1 C(C(=O)NCCCOCCCCN(C)C(c1ccn(C)n1)C)(C(C)C)OC C1(NC(c2n(C)c(=O)ccc2)=O)CCC2(CC1)CCN(C(=O)CC1CC(F)C1)C2 CCC(C)C(C(=O)OC)N(C(=O)C(C)CCOC1CCN(C)CC1)C C1(NC(c2ccc(C(N)=O)o2)=O)COCCC1NC(=O)C(O)c1ccsc1 c1(OC)ccc(C)c(NC(=O)C(Cc2cn[nH]c2)NC(=O)CN2CCC(C)C2)c1 Cc1ccc(C(N2CCC(O)(CCNC(=O)C(C)n3cncn3)C2)=O)n1C N1(C(Cc2c(C)nc[nH]2)=O)CCN(C)CC1CNC(c1cc(N)cnc1Cl)=O Cc1cc(N)cc(C(=O)NCC(CNC(C2CCCN2C)=O)CO)c1F COn1cnc(C)c1C(=O)NCC12CCC(CO)(CC1)O2 C(=O)(C1Cc2ccccc21)N1CCC(NC(C2(C)CC=C(C)CC2)=O)C1(C)C C(=O)(C(C)CNC(=O)CCC=CC(C)C)N(CCCC#C)CC C[Si](C)(C)c1cccc(-c2noc(C3CC34CCC(F)(F)CC4)n2)c1 c1(C(=O)NCCCC(C)NC(C2CSCCS2)=O)c(Cl)c2ccccc2n1C C1(C(=O)NC2CCC(NC(COc3c(C)cccc3)=O)CC2)CC2CCC(C1)C2 c1(CNC2CN(C(c3cnc(O)c(Cl)c3)=O)CC(F)C2)c(F)cc(Cl)cc1F C#CCCCCCCC(=O)NC1CCC(C)N(C(c2cnc(C(C)=O)s2)=O)C1 C(=O)(CCC(C)(C)C)NC(C1CCCN(c2nnc(-c3ccccc3)s2)C1)C CC1CCC(=CC(=O)NCc2cnn(CC(=O)N(CCC(C)SC3CC3)CC)c2)C1 N1(CC(CC)NC(C2CC(n3cc(COCC)nn3)C2)=O)CCCCCC1 c1(C(N2C(C(N(CC(C)(C)CO)C)=O)CCC2)=O)ccc(CSC)cc1 C1(C)(CNC(CC2CCN(C)CC2)=O)CN(c2ccncn2)CCO1 C1(NC(c2c(C)cc(C)s2)=O)CCN(C(=O)CCCn2ccnc2)CC1C(N)=O c1(C(C)C)cc(C(N2CC3C(CNC(C4CCOC4)=O)C3C2)=O)n(C)n1 N1(C(c2cc(SC)c(C)o2)=O)CC2CCC1C(CNC(C1CCCCC1O)=O)C2 c1(C(=O)NC2C(C)N(C(c3csc([N+](=O)[O-])c3)=O)CCC2)cccn2cnnc12 c1(NC(C2C(C(=O)OC)C2)=O)cc(Cl)ccc1C(=O)Nc1ccc(Br)cc1O c1(C(=O)NC)cccc(C(N)=O)n1.C(C)(C)(C(=O)NCCC1(C(=O)N)CC1)SC O(NC(=O)C(C)NC(c1ccc(C(C)C)o1)=O)C(C=C)C c1(CSC)ccc(C(=O)NCC(C)(C2CC2)NC(=O)CC2CCC(F)(F)C2)cc1 C1(C2(O)CC2NCC(O)CO)CCCCCC1 CC1CCCCN(C(C2CNC(=O)CN2C(=O)Cn2ccccc2=O)=O)C1 c1(N(CC(=O)NCCNC(C(C)C#N)=O)C)nccc(NC2CC2)n1 C12(OC)CCC(C(=O)NCC(C3CCC3)NC(=O)CC=C(Cl)Cl)(CC1)C2 C1(O)(CN(C(Cc2cc(C)no2)=O)C)CCN(C(c2ccccc2Cl)=O)C1 C1(CNC(c2nn(C)c(F)c2)=O)CN(C(C2SCCS2)=O)C2CCN1C2 C1(CNC(COCc2ncc(C)o2)=O)CC2(CC2)CN1C(C1CCC1C(F)F)=O C1(C(N(C(C#C)C)C)=O)CCCCCN1C(c1[nH]ccc1COC)=O C1(C(N(CCN(C(C)C)C(C2CC2c2cncs2)=O)C)=O)CC12CCCCC2 C1(C(=O)NC(CNC(c2c(C)oc(C(C)C)c2)=O)C)CCCNS1(=O)=O N1(C(c2cc(F)cs2)=O)CC(NC(C2(CO)CC2(F)F)=O)C(O)C1 c1(C(=O)N(c2nc(C)c(C(=O)N(C)CC#N)s2)C2CC2)ccc2c(c1)CCC(=O)N2 C(=O)(C1=CC(C)(CC)C1)NC1C2CN(C(c3c(OC)scc3)=O)C1C2 c1(CN(C2CCCC2CN2CCC(NCCO)CC2)C)ccc(Cl)c(Cl)c1 c1(C(=O)NC2CN(C(c3cn(CCOC)nc3)=O)C2)cc(C)n(C(C)C)n1 N1(C(C(CC2CC2)OC)=O)CCN(CC(C)(C)NC(=O)CCC2CC2CN)CC1 c1(C(N2CC(CN=c3cc(C)nc[nH]3)OCC2)=O)cnc2ccccc2n1 CC1(C)CC(C)(NC(=O)COC2CC2(F)F)CN1C(c1cnn2cccnc12)=O CC1CCCn2ncc(CN3CCC(NC4CCCNC4=O)CC3C)c21 C1(CNC(C=C(CCC)C)=O)CN(C)CCN1C(C1CC1CCOC)=O C(C(=O)N=S1(=O)CCC2(CCCN2)C1)c1cccc(N(C)C)n1 C(=O)(CCC(C)S(C)(=O)=O)NC1CCN(C(C=C(C)c2cccc(Br)c2)=O)C1 C(C1CCCC1)=C(C)C(=O)NCC1(O)CN(C(=O)C=CC(=O)NC2CC2)C1 C1(F)(CNC(CC2(N(c3ccc(F)cc3)C)CC2)=O)CCN(C(c2cnns2)=O)C1 N1(C(C(=Cc2ccncc2)C)=O)CCC(CO)(NC(C2CC(O)C2)=O)CC1 Cc1cc(C(=O)NC2CC(NC(=O)CC(O)CF)CC2O)c(Br)cc1F C1(NCc2c(O)cc(Cl)cc2)CCCC12CCCO2 C(C(=O)NCC1CC(NC(=O)CCCC(F)(F)F)C1)(C(C)C)(C(C)C)NC(C)=O c1(C(=O)NCC(C2CCN(C(C3CCSC3)=O)C2)(C)C)c[nH]nc1[N+](=O)[O-] c1(CC2CCN(C(c3c(C)[nH]cc3C(=O)O)=O)C2)cccc([N+](=O)[O-])c1F C(=O)(CCCCCCN=[N+]=[N-])NCC(CC(C)C)NC(=O)C(C)CCN(C)C C(CN=c1[nH]n2cc(C)nc2s1)NCCNC(C(CCCOCC)C)=O N1(C(C2(Cl)C(C(C)=O)C2)=O)CC2(C1)CN(C(=O)COC1CCOCC1)CCO2 Cc1cc(Cl)nc(Cl)c1C(=O)NC1CN(C(c2cnnc(O)c2)=O)C1 C#Cc1cncc(C(=O)N(CC(C)NC(c2cnc(-c3ccncc3)s2)=O)C)c1 CC(C)(C)CCC(F)C(=O)NC1CC2(C1)CC2NC(=O)Cc1cccc(C#N)c1 c1(C2(C(n3ccnn3)NC3C(C(=O)OC)C3)CC2)ccc(Cl)cc1 c1(C(N2CCN(C(=O)NCC3CCCCC3(F)F)CC2)=O)cn2c(n1)SCC2 C1(NC(CCCc2scc(C)n2)=O)CCN(C(=O)COc2ccon2)CC1O C(=O)(C(C)(C)CCN(C)C)NC(CC)CNC(=O)C(C)(C)CSC N1(C(C2(C(F)F)CCOC2)=O)CCOC(CNC(C2CC(=C3CC3)C2)=O)C1.CCOC c1(C(C(=O)N(C(CC(=O)OC)C)C)(C)C)ccc(Br)c(Cl)c1 CC1(CNC(=O)Cc2cnc(C3CC3)[nH]2)CCN(C(C2(F)CCOC2)=O)C1 c1(C(n2cc(C(C)(C)NC(Cc3c(C)nn[nH]3)=O)nn2)C)ccc(Cl)cc1 n1(CC)ncc(C(=O)OCC2CCCC2C)n1 C(=O)(C(C)CS(C)(=O)=O)NC(CN(C(C(C)CC1CC1)=O)C)(C)C C(=O)(C1=NOC2(CCC2)C1)NC1C(CC)N(C(c2cc(F)n[nH]2)=O)CCC1 CC1CCOCC1C(N1CCC(C(C)(C)C(=O)NC(C)(C)CF)C1)=O N1(CC(=O)N(C2CN(C(=O)CC34CCCC3C4)CC2F)C)CCCCC1=O CN1CC(C)(C(N2CCCCC(C(=O)NC3CC(=O)N(O)C3)C2)=O)CC1=O c1(OC)cc(NC(=O)C(c2ccc(CC(C)C)cc2)C)c(Br)cn1 Cc1cccc(C)c1C(N1CCC(CN(C)C(c2cc(Br)c[nH]2)=O)C1)=O N1(C(C2N(C)CC(O)C2)=O)CC(NC(=O)CCc2ccc(F)cc2Cl)C(C)(C)C1 c1(C(N2CCC(CN(C)CC)C2)C(=O)NC(CC)C)ccc(Br)c(F)c1 N1(C(C2CC3CCN(C(c4cc5ncccc5[nH]4)=O)CC32)=O)CCC2(CCSC2)C1 C1(C(=O)NCCNC(C(c2ccc(C(F)(F)F)cc2)CC)=O)CCCC1(C)C c1(CC(=O)NC(C)CCN(C(=O)C(C)C2CCC2)C)cccc(Br)c1F CCCC(C(O)C(=O)NC(C)(C)C(C)O)NC(C(C(=O)OC)C(C)C)=O Cc1cc(CC(=O)NCC2CCCC2CNC(=O)CN(C)S(N)(=O)=O)cc(C)n1 C#Cc1ccc(C(N2CCC(CNC(C3(C4CCC4)CC3(F)F)=O)C2)=O)c(F)c1 CCC1=NOC(C(C2CCN(C(C(C3CC3)NC34CC3CNC4=O)=O)CC2)N(C)C)C1 c1(C(N2CC3C(CNC(c4ccc[n+]([O-])c4)=O)(C3)C2)=O)cc(Br)cnc1F C1(CC(=O)NC2(C(=O)NCc3nnc(CC)o3)CSC2)CCCC2CC12 N1(C(CCOCC)=O)CCN2C(=O)C(NC(c3nccc(Cl)c3F)=O)CC2C1 C1(C(=O)NCC(C)(F)Cl)(NC(c2cc(C(C)C)no2)=O)CCN(C)C1 C1(CNC(C2CN(C(C3(C4CC4)CC3)=O)CC2C=CC)=O)Cc2nccn2C1 C1(NC(C(C)SC)=O)C2CCN(C(=O)CNC(c3cnccn3)=O)C12 N1(C(c2[nH]cc(C)c2)=O)CCC2(NC(c3cc4n(c3)CCC4)=O)CC2C1 C1(CNC(c2nc(C)oc2)=O)CN(c2ncc(F)c(-c3ccsc3)n2)CCCO1 N1(C(CC(CC(C)C)C)=O)CC23CCCC2(C1)CN(C(=O)CCc1nc[nH]n1)C3 N1(C(c2cc(C)on2)=O)CC2CCCC(N(C(=O)CC(C)C(F)F)C)C2C1 CCCC(O)(CCC)CC(=O)NCC1CN(C(=O)C(F)(F)CC2CC2)CC1C c1(C(C(=O)Nc2oc(OC(F)F)nc2-c2ccccc2)SC)ccc(Cl)c(Cl)c1 C12(C(=O)NCC3(NC(c4ccc(CCC)[nH]4)=O)CCC3)C3CCC(CC13)C2(F)F C#CCCCCC(=O)NC1CCCCCC1NC(c1cnn(C(F)F)c1)=O N1(C(CC2(COC)CC2)=O)CC2OCCN(C(=O)Cn3cc[n+](C)c3)C2C1 c1(C(N2C(CNC(CSCC=C)=O)CC2)=O)cn(C)c(=O)nc1O CCCCC(=O)NC.C1(O)(C(=O)OC)CC(C(=O)NCC2C(C(=O)OC)C2)C1 C(C)(CCC(=O)N(C(C)CNC(c1cc(C#N)c[nH]1)=O)C)OC C1(C(=O)NCC(CNC(=O)Cc2ccon2)F)CCc2nncn2CC1 C1(C(=O)NC2CCCN(C(C=CC3N(C)CCC3)=O)C2)Cc2cscc2C1 Cc1onc(-c2ccccn2)c1C(=O)NC1CC(CNC(c2csc(Cl)n2)=O)C1 c1(NC)cccc(C(=O)NCC(C(C)(C)C)NC(C2(CS(N)(=O)=O)COC2)=O)c1 C1(NC(c2c(Br)cn(C)n2)=O)CCN(C(c2ns[nH]c2=O)=O)CC1CO N1(C(COCCCC#C)=O)CCC(CNC(c2cscc2OC)=O)C(C)C1 C1(CC(=O)NC(C(C)C)CNC(=O)C(F)CC(C)(C)C)CC(C)(C)OC(C)(C)C1 Cc1c(C(N2CCC2CNC(=O)C(C)(F)F)=O)sc2ccc(Br)cc12 c1(C(=O)NCCC(CNC(C2(C=C)CCOCC2)=O)=C)ccc2ccncc2c1 C1(C(=O)NC2CC(CCOC)C2)CCOCC1NC(c1cc(F)n(C)n1)=O c1(OC)cncc(C(N2CCC(C(=O)NCCN(C)C)C2C(C)C)=O)n1 N1(C(c2cc(CC)on2)=O)CCCC(N(C)Cc2cc(C)nn2C)C1 c1(OCCCOC)ccccc1C(=O)NC(C)CN(C)C(c1c[nH]c(CO)c1)=O C=CC(C)(O)C(=O)NCC1(COC)CCCC1.c12cn(C)nc1NC2=O CC(C(C)(C)NC(=O)CCOCC1CC1)NC(c1cc(-c2ccccc2)cs1)=O c1(CNC(c2cccc(CC)n2)=O)ccc(CNC(=O)C(F)C(C)(C)O)c(F)c1 C#CC(CC(C)(C)C)NCc1cc(-n2ccnc2C)ccc1C c1(CC(=O)N(C(C)C)CCNC(=O)C(O)C(F)(F)F)ccc2ccoc2c1 N1(C(C(C)=C2CC2)=O)CCC2(CC1)CC2CNC(=O)CCc1cccnc1F c1(NC(=O)NC2CCCC(CF)C2)ccccc1C1CCCC1 Cc1nnc(NCC2C(C)CCCN2C(C2CC2(C)C)=O)c(C#N)c1C O=C(CC1OCCc2ccsc21)NC1CN(C(=O)CCc2cncs2)CC1F C1(C)(CCC(=O)NC(c2n[nH]c(CO)n2)C)CN(C(c2ccn(CCF)n2)=O)C1 C=CCN=C(NCC(C)C(F)(F)F)NC1CC(OCC)C1.C(C)(C)(C)O N1(C(C)C2CC2c2ccccc2Cl)CC2CCC(C1)C2O.Cc1ccsc1-c1ccn[nH]1 c1(OCC)cccnc1.C1(C)C(=O)NC(C2CC2)CNC(=O)C=CCN1C C1(OC)CN(C(=O)NC2CC(F)(F)C2C)CCC1(CO)OC c1(NC(C2(N)CCC(CC)C2)=O)ccc2c(c1)OCC2 CCC(CC)C(C(=O)NC(C)CC(C)NC(c1cc([N+](=O)[O-])nn1C)=O)OC C12(CNC(C3(CCCC)CC3)=O)CCC(CN1C(c1cc(C)ccc1F)=O)C2 C12(C(=O)NCC(CNC(CCC(=O)N(C(C)C)C)=O)(C)C)CC1COC2(C)C Cc1ccc2ncc(C(=O)NCC(F)CNC(C3CCCN(C)C3)=O)n2c1 Cc1cncc(C(=O)NC(CNC(c2ccc(N(C)C)cc2)=O)C(C)C)c1C C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(CNC(n2ncc(C)c2)=O)(C)C)C1 c1(C(=O)NC2CCN(C(C3(C)CNC(=O)C3)=O)C2)nnc(O)c(Br)c1O Cc1cc(C(N2C(C(=O)NCCC3(O)CCCC3)CCC23CC3)=O)c[nH]c1=N C1(C(N2CC(C)C2(C)C)=O)CN(C(C2CCC(C#N)CC2)=O)C(C)(C)C1 Cn1ncc(C(N2CCOCCC2c2ccc(C(F)(F)F)cc2)=O)cc1=O N1(CC2(C)CCOCC2)CC(=O)N(Cc2csc(Cc3ccsc3)n2)C1=O N(C1CCc2cccnc21)C(C1(C)CC(NC(c2cc(C)sc2C)=O)C1)=O C(C(C)(O)C(=O)N1CCOC(CNC(C2NC(=O)CC2C)=O)C1)OC Cn1nncc1C(F)(F)C(=O)NCC(O)CNC(C12CC(F)(C1)C2)=O C(CCC(C)C)(C(=O)NC1CCN(C(C23COCC(C2)C3)=O)CC1F)NC(C)=O N1(C(CNC(c2cc(OC)ncc2)=O)=O)CC2CN(C(c3ccco3)=O)CCC12 N1(C(C2CCN(C(CC)=O)C2)=O)CCC(F)(CNC(C2CCOC2(C)C)=O)CC1 N1(C(c2ccc[nH]2)=O)CCN(C(C2(n3cnnn3)CC2)=O)C(c2ccccn2)C1 Cc1cc(C(N2CCC(CC(=O)N(C)Cc3cccc(O)c3)C2)=O)ncc1CO c1(CC(=O)N(C(C(=O)NCCC(O)C2CCCC2)C2CC2)C)cc[nH]n1 c1(CNC(=O)OC(C)(C)C)ccn2cccc2c1.C12CCCCCN1C2=O Cc1cc(C(=O)NCCC2CN(C(c3c[nH]cc3C(C)(C)C)=O)C2)cc(C)n1 CC1(CO)CCN(C(C2CCN2Cc2cc(Br)c[nH]2)=O)CC1O C1(C(=O)NCCCNC(c2n(C(C)(C)C)ncc2)=O)C2CCCCCCC12 c1(C(=O)NC(CC)CNC(c2ccc([N+](=O)[O-])s2)=O)cc2cc(F)ccc2o1 CC1(C)CCC(C(=O)NCCCC2CN(C(c3cc(C#N)c[nH]3)=O)CCO2)C1 C1(n2cc(-c3ccc(C)cc3)nn2)CCCN(C(=O)Nc2cc(Br)cnc2F)CC1 N1(C(CCOCCOC)=O)C2CCC1C(C(=O)N(CC(O)COC)C)C2 C(c1cscn1)=CC(=O)NC1CC(CNC(C(C)NC(C2CCCC2)=O)=O)C1 O=C(CCC1CCc2ccccc21)NCC1(CNC(C23CC(F)C2C3)=O)CCC1 c1(C(=O)NCCCC(C)NC(=O)C=Cc2cncn2C)cc2cccn2c(O)n1 c1(C(C)C(=O)N(CCCF)C)ccccc1-n1cc(CN(C)C)nn1 CC1(C#CC(=O)NC2CCC(NC(=O)CCCC(N)=O)CC2)CC1 c1(OC)ccc([N+](=O)[O-])c(N2CCC(CCNC(=O)CCN3CCCCC3)C2)n1 CCCCC(CC)CC(=O)NC1COCC1NC(=O)C=Cc1cccc(C)c1 N1(C(c2c(CC)n(CC)nc2)=O)CCC(NC(c2csc(CC)n2)=O)CC1C c1(OC)cccc(Br)c1C(C)Nc1nccc(NC(C2CCCC2)C)n1 c1(C(=O)NCC2CC2NC(c2nncn2C2CC2)=O)cc(-c2ccco2)c[nH]1 C(C1=CCCN(C(=O)C=CC(C)C)C1)NC(C(COCC)C)=O C1(CNC(c2cc(CC)c(CC)o2)=O)CC2(CC(NC(=O)C(C)(C)CF)C2)C1 Cn1ccc2c(C(N3CC(NC(=O)C(O)C4CCC4)CC3(C)C)=O)cnc(O)c12 C1(C(=O)NCC2CCC(CC)CC2)CCCCC1NC(=O)CSC(F)F C(N=c1[nH]c(=NCCC2CCC2)[nH]c2c1CCCCCC2)C1(C)NC(=O)NC1=O C1(NC(C(c2ccnn2C)C)=O)COCCN(C(=O)CCC(C)N(C)C)C1 C1(C(=O)NC(C(C)NC(=O)CN2CSCC2=O)C)CC(F)(F)C1(C)C C(CCCCC(=O)NC1CC(C(=O)N(CCC(=O)OC)C2CC2)C12CCC2)=CC C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1OCCN(C(c2cccc(C)n2)=O)C1)C N1(C(c2c(CC)nc(C)[nH]2)=O)CC2N(C(c3nc(C)ccc3F)=O)CCC2(C)C1 c1(NC)ccc(C(N2CC(CNC(C34CC(O)C3C4)=O)C(C)C2)=O)cc1F Cn1cnc(COC(=O)CC2(C)CC2(F)F)c1 C1(CC(=O)NC2C(C)CCN(C(C3CCC4CC4C3)=O)C2)Cc2ccccc2N1 C1(NC(C(CCSC)(C)C)=O)CC2CC1CN(C(c1cc3cn[nH]c3cn1)=O)C2 N1(C(c2c(C)cn(C)c2)=O)CCC(NC(=O)COc2cccc(F)c2Cl)C(O)C1 C1(C(=O)NCC2CCOC2C(C)C)(CC)CN(C(=O)COCCC(C)C)C1 Cc1nc2cc(CN3CCC4CN(C(c5cncc(F)c5)=O)CCC34)ccc2o1 c1(C(=O)NC2CCN(C(C3C(C)(C)CO3)=O)C2C2CC2)cnc2cc[nH]c2c1 CCCCC(=O)NCC(C)C(=O)NCCC1(C)CCOC1 c1(C(=O)NCC2CCC(NC(CSCC(N)=O)=O)C2)nccn2nccc12 N1(C(CC(CC)(F)F)=O)CCN(C(=O)C(C)c2ccsc2)CC2CCCCC12 c1(C(=O)NC2(C(=O)NC(CC#CC)CO)CC2)ccc(C)c(O)n1 O(NC(=O)C(C)(C)O)C(C1CC1(C)C)C.C(C(=O)OC(C)(C)C)NC(=O)OC(C)(C)C n1(CC)ncc(C(=O)NCC2CCN2C(C2(C)CC(C)C2)=O)n1 C1(C(=O)NC2CCN(C(CCC=C(C)C)=O)C2C)CCn2c(C)nnc2C1 CC#CCC(C(=O)N1CCC(COC)C1)NC(C1(OC)CCOC1)=O N1(C(C2CC(=C)C2)=O)CCC2CCN(C(C3CCc4nc(C)cn4C3)=O)CC2C1 N#CC12CC(C(N3CC(NC(c4cc(C5(O)COC5)on4)=O)C4CC34)=O)(C1)C2 CS(=O)(=O)CCCNC(c1nnnn1CCCSCC#N)(C)C1CC1 c1(C(N(C(CCNC(C(C)c2cccs2)=O)C)C)=O)ccn2nncc2c1 c1(OCC(=O)NCC(C)NC(C2(c3ccnn3C)CC2)=O)cnn(C)c1 c1(OCCN(C)C(=O)NC2CCCN2CC2(C)COC2)ccc(S(N)(=O)=O)cc1 c1(NC(c2c(SC)csc2)=O)ccc(NC(c2cc[nH]n2)=O)c(C)c1 Cc1ccc(O)cc1NC(c1cncc(-c2cn(C)nc2C)c1)=O c1(CNC(Cc2nc(C)[nH]n2)=O)cccnc1CNC(C1COCCN1C)=O c1(COC(C(=O)NC(CN(C(C2C(C)CCC2)=O)C)(C)C)C)ccc(Cl)cc1 N1(C2CCN(C(C3C(C)C3)=O)C2)CCC(NC(=O)COc2cnn(C)c2)CC1 CCC(CNC(C1(NC(c2c[nH]c(=N)o2)=O)CC(O)C1)=O)CC(C)C c1(C(=O)NCC2CCC(C)CN2C(c2ccns2)=O)cc2sccc2cn1 N1(C(c2ccn(CCC)n2)C(=O)NC(C)C)CCOC(Cc2ccccc2)C1 CCCC(C(=O)NCC1(F)CC(CNC(=O)CCSCC(C)C)C1)OC C(=O)(C(CC(C)C)OC)NC1(CC(NOCC)=O)CC1.C1(=O)CCCN1 C(C1=CCN(C(c2ccns2)=O)CC1)NC(=O)Cn1cc(C2CC2)cn1 CCC(C)C(C(=O)NCCC1(NC(=O)Cc2ccc(C)nc2)CC1)OC C(C(C)=CC(=O)NC1(CC(=O)NCCCOC2CC2)CC1)OC O=C(CCC(CF)CF)NC1CCC1NC(c1nccc2occc12)=O c1(CC)cc(Cl)ccc1C(=O)NCCCC1(NC(c2cnc(C)o2)=O)CC1 Cc1noc(Cl)c1CC(=O)N(CCCN(C)CC=CC(C)(C)C)C C1(CC=C)(NC(=O)CSc2ncccn2)CCN(C(=O)Cc2cccnc2F)C1 N1(C(CC(C)c2ccco2)=O)CCCC(O)(CNC(c2cn3ccnc3s2)=O)C1 c1(C(C)C(=O)N(C2CC(NC(c3cnns3)=O)C2)C)cccc(O)c1 CC(C)(C(=O)NC(c1ccccc1)CNC(c1ccc(C(F)F)s1)=O)C(F)(F)F Cc1nc(O)[nH]c1C(=O)NCCCOCCNC(c1ocnc1C)=O N1(C(CC2CCC(C)O2)=O)CCN(C(c2cnn(C)c2)=O)C(CCO)C1 CC(C)(C)CC(CO)NC(c1coc(CNC(=O)C(O)CC(N)=O)c1)=O Cc1cc(CCC(=O)NCC2CCN(Cc3ccsc3)C2)no1 c1(C(=O)NCC2C(C)(C)C(NC(C3CS(=O)(=O)C3)=O)C2)cn2cccnc2n1 C1(CC)CCN(C(c2nnc(S)n2C)=O)C1C(=O)NCCCC(N)=O c1(C(N2C(C(=O)Nc3cccc(O)c3)CC2)=O)cc(Br)cnc1O C(c1ncccc1C)=CC(=O)NC(CNC(C1N(C(C)=O)CCCC1)=O)C(C)C C1(CNC(CNC(C2CCN(CC(C)C)C2)=O)=O)CN(C(C)C)CC1C C1(C)(CNC(C2(CCC)CC2)=O)CCCN1C(c1sc(C)nc1C)=O CC(C)(F)CCC(=O)N1CCC(CNC(c2ncnc(O)c2F)=O)C12CC2 CCC(CC)C(CNC(c1cn(CC2CCCO2)nn1)=O)N1CCOCC1 c1(C(c2n(C(C)C)nnn2)NCC2COC(=O)N2)cc2c(Cl)nccc2s1 Cc1sc(S(N)(=O)=O)cc1C(=O)N(CC(C)N(C)C(c1ncncc1F)=O)C Cc1cc2c(cc1C)OC(CNC(=NCCCOC1CCOC1)NCC1CC1)C2 c1(C(=O)NC2C(NC(c3ccc(C)s3)=O)CC2)cccc(C2CC2)c1Cl C1(C(=O)NCC2C(F)(F)CCN(C(C(C(C)C)O)=O)C2)CCC(C2CCCO2)O1 Cc1nc(C)c(C(=O)NCC(C2CC2)NC(c2cncc(-n3cccn3)n2)=O)s1 C1(NC(c2csc(O)n2)=O)CC(O)CN(C(c2ccc(=O)oc2)=O)C1 c1(C(=O)NCC(=C)CCNC(C2CC2(C)C(F)F)=O)cnc2n1CCOC2 C1(CCOC)CN(C(c2ccnn2C(C)CC)=O)CCN1C(=O)Cc1cnns1 C12CCN(CC13CC3)C(=O)N2.C1(CS(C)(=O)=O)(N(C)C(=O)OC(C)(C)C)CCC1 c1(C(N2C(CNC(c3n[nH]c(CC)c3F)=O)CCC2)=O)c(Br)ccc2c1OCO2 C1(C(C)(C)C)CCCC(C(=O)NC(=O)NOC(c2cccs2)C2CC2)N1 C1(CNC(CCCCSC)=O)CC(C)(C)CN1C(=O)Cc1sccc1Cl C(=O)(C(CC(C)SC)N(C1(C#N)CCC1)C)NC(CC)CC c1(C(=O)NC2CCC(NC(CC(C)SC)=O)CC2)ccc2c(c1)N(C)C(=O)CC2 c1(C(N(CC(C)N(C(c2c[nH]c(=NCC)s2)=O)C)C)=O)cccc(S(N)(=O)=O)c1 Cc1ccc(C(C)C)c(C(N2CCC(CNC(=O)C3=CC(C)C3)CC2)=O)c1 Cc1cc(F)cnc1C(N1CCC2(NC(=O)CC3(N(C)C)CCCC3)CC2C1)=O Cc1ccc(O)nc1CNC(=O)C=CC(C)(C)NC(c1c(C)coc1C(C)C)=O c1(C(=O)NCC(CC=C)NC(=O)C(O)CC[S+](C)C)cc(Cl)c(N)cc1F N1(C(C=Cc2c(C)nccc2)=O)CCCC2C1CCCN2C(c1cn[nH]c1)=O Cc1c(Cl)ccc(C(N2CCC(F)(CNC(=O)CC(C)N(C)C)C2)=O)c1O CC1CC(NC(=O)CC23CCC(CC2)C3)CN(C(c2cn(CCO)nn2)=O)C1 c1(C(N2CCC(CN=[N+]=[N-])C2)C(=O)NCCCC)cccc(Cl)c1OC Cc1c(NCCC(=O)N2CCCC2)ncnc1NC1CCOC1C CC1(CCC(=O)NC2C3CC2N(C(=O)CN2CC4CC4C2)C3)CCC(=O)N1 c1(C(=O)NCC(CNC(c2c(C)nc[nH]2)=O)C)ccc(C(=O)OC)c(O)c1 N1(C(c2nnc(C)o2)C)CC(NC(c2sc(C)nc2C)=O)C(C)(C)C1 c1(C(=O)NCC2(NC(c3cc(N)c(Cl)cc3)=O)CC2)cc2nn[nH]c2cc1F c1(C(=O)NCC(CC)NC(=O)COc2cccc(F)c2F)c(C#N)cnn1C n1(C(C)C)cnc(C(N2CCC2CC(=O)NCC2CC=CCC2)=O)c1 CC1CC(CNC(=O)C(F)n2cccn2)CN1c1ccc(C(N)=O)nn1 c12ccc(o1)SC(C)CN(C)C(=O)C1(CCC1)N(C)C2=O.N1(SC)CCCCC1 N1(C(Cc2cc(C)cc(C)c2)=O)C2CCC1CC(NC(c1cnn(CO)c1)=O)C2 C12(C(N3CC(CO)C3)=O)CCCC1N(C(=O)C(COCC)OC)CC2 CCCC(C(=O)N(CC(CC)NC(C1(CF)CC(F)(F)C1)=O)C)N(C)C C1(NC(CCNC(COC)=O)=O)CN(C(c2csc(=N)[nH]2)=O)CC12CCOCC2 c1(N)snc(Cl)c1C#N.c12cc(on1)C(=O)NCCCN2C(C)C.C1CC1 n1(CC(=O)NCC2CN(C(COCc3n(C)ccn3)=O)CC2O)ccc(O)nc1=O C(CC(C)C)(C(=O)NCc1cn(CCO)nn1)ONC(c1c(C)nsc1N)=O C1(C(=O)NC2C(C=C)CN(C(C3OCCC3(C)C)=O)C2)CCCC(C)(C)CC1 N1(C(c2scc(C#N)c2)=O)CCC(O)(CNC(C2CCS(=O)(=O)C2)=O)CC1 c1(C(=O)NCCN2CCN(C(C=CC=CCC)=O)CC2)cccc(C#CCO)c1 C1(NC(=O)C=Cc2cccs2)CC(F)CN(C(=O)Cn2cnnc2)C1 CCCCCCCCC(c1nnnn1C(C)(C)CC)NCc1ccc(F)cc1Br c1(C(=O)NC(C2CCN(C(c3c(C#C)c[nH]n3)=O)C2)C)nn(C)cc1[N+](=O)[O-] c1(C(N2CC=C(C#N)CC2)C(=O)Nc2ccc(OC)cc2)cc(F)cc(Br)c1 c1(C(=O)NCCC2OCCN(C(C(CCC)OC)=O)C2)c(F)cc(C#N)cc1F C(=O)(CC(O)C(Cl)(Cl)Cl)NC(C)CCNC(c1cnn(C)c1C(F)F)=O NS(=O)(=O)c1cccc(C(=O)NC2CN(C(=O)CO)CC2O)c1 C(=O)(CC(C=C)CC)N(CC(=O)OCC)CC#C.C(CO)(C1CCC1)C C1(NC(C2N(Cc3ccc(N(OCC)CC)o3)CCC2)=O)CCNC(=O)CC1 N1(C(C(CCC)(C)CC)=O)CC2CCC(NC(=O)C(CC)N(C)C)CC2C1 C(=O)(CC1CCc2ccccc21)N(CCNC(c1ccc(N)c(C)c1C)=O)CC N1(C(C2CCCN(C(CC)=O)C2)=O)CC2CN(C(=O)C3=NOC(C)(C)C3)CC2C1 c1(C(=O)NC(CCNC(C(C)NC(C)=O)=O)(C)C)cn2cccc(Cl)c2n1 CC1(C)OCCC1CC(=O)NC1CC(NC(c2ccnnc2O)=O)C(O)C1 CC1(C)CCCOC1C(N1CCCCCC1C(=O)NC(CCO)C(C)(C)O)=O C1(CN(C(C(CC)n2nccc2C)=O)C)CCCCN1C(c1nc(Cl)cs1)=O c1(C(=O)NC(CC)(CNC(c2cccc(N)c2)=O)CC)cc2nc(Cl)ccc2s1 N1(C(c2cncc(NCC)c2)=O)CC(O)C(O)C1CNC(c1ccnnc1)=O S(=O)(=O)(CC(=O)NC(C)C(C(C)C)NC(c1cc(CC(C)C)nn1C)=O)NCC c1(CC)cnc(C(N2CCC(C)C2C(=O)N(C)Cc2nc[nH]n2)=O)nc1 N1(C(N(C)CC)=O)CCC(O)(C(=O)NCCSCC)C1 c1(C(N2C(C)CC(NC(C3(CC#C)CCCC3)=O)C2)=O)cc(Cl)cc(F)c1N CCCCC(C(=O)NCC1CC(NC(=O)CC2OCCO2)C1)NC(N)=O c1(NC(N(CCC)CCN(C)C)=O)ccc(OC(C)CC)c(Cl)c1 c1(C(N(CC(C)NC(=O)C(COC)OC)CC)=O)ncc(Br)cc1N C1(C(C(N2CC(=CC)C2)=O)NC(=O)CSc2cn[nH]c2)CC=CCC1 N1(C(C(CC)F)=O)CCN(C(=O)C(C)N(C)C)CC1CCO c1(C(N2CC(C)CC(NC(c3ccc(CC)s3)=O)C2)=O)cccc2[nH]ncc12 C=CCC(C(=O)NC(C)(C)C)NC(=O)NC1CCCN(CC(=O)OC)C1 C12(C(N3CC(N(C(C(CC)CC=C)=O)C)C(C)(C)C3)=O)CCCN(C1)S(=O)(=O)C2 c1(NCc2nnn(C(C)(C)C)n2)nccc(=NCc2cccc(C(F)F)c2F)[nH]1 Cc1c(C(N2CCN(C(C3COC(=O)O3)=O)C(C)C2)=O)oc2ccccc12 c1(C(=O)NCC2C(NC(c3c(C)cn(C)n3)=O)C2)cc(F)cc2cccnc12 c1(OCC)cccc(CC(=O)NCC(O)CNC(=O)CCn2ccnc2)n1 CC1CN(c2ccnc(NCc3ccc(O)nc3)n2)CC1CS(N)(=O)=O C1(NC(=O)CC2CCCOCC2)CCCN(C(=O)CCCn2cccn2)CC1 Cc1ccn2c(C(=O)NC(C)CN(C)C(c3nc(O)sc3C)=O)cnc2c1 c1(CNC(c2n(C)cc(Br)n2)=O)ccc2[nH][nH]c(=N)c2c1 Cc1cc(NC(=O)C(C)OC(=O)Cc2cscn2)ccc1C(C)C C1(=O)C(CC(C)C)O1.C1(NC(C(c2ccc(F)cc2)SC)=O)CCCC(C2CC2)O1 C(c1ccc(Cl)s1)=CC(=O)NCCOCCN(C(C1(C(C)C)CC1)=O)C N1(C(C(C2CN(C(CC(C)(C)C3CC3)=O)C2)O)=O)CC2CCC(C1)C(=O)N2 C1(N(CCCCN(C(=O)Cc2ccco2)C)C)CC(=O)N(CC2CC2)C1=O C1(NC(c2cc3c(nn2)CCCO3)=O)C2CC3CN(C(C4CC=CC4)=O)C1C3C2 c1(OC)ccc(C)cc1C=CC(=O)NC(CCN(C)C(C1(C)CC1)=O)C(C)(C)C c12ccc(c([N+](=O)[O-])c1)N1CC(C1)NC2=O.c1(C(CC)(F)F)ccccc1 C(=O)(C(CC#CC)NC(=O)C(C1CCOCC1)F)N1CC(C#C)(N(C)C)C1 C(=O)(C(C(C)C)SC1CC1)NCCC1(C(=O)NC2(SCC)CC2)CC1 C1(NC(c2nccc(C)c2)=O)CC2CN(C(=O)C(C)C3CCOC3)CC12 C(=O)(NNc1cccc(C)c1F)C1CC2(CCN(Cc3c(C)nn(C)c3)CC2)C1 c1ccc(C(C)O)cc1.C1(C(N(CCN(C=O)C(C)C)C(C)C)=O)CCCN1N=O C(C)(C)(CCCNC(c1cn(-c2ccc(C)cc2)nc1C)=O)NC(C(CC)C)=O c1(CC(=O)NC2CCC2)ccccc1-c1cccc(C2CC2)c1 N1(C(C=CC)=O)CCC2(CCCCN(C(=O)COCC3CCCCO3)C2)C1 C1(NC(C2N(C)C(=O)CCC2)=O)CN(C(c2cnn[nH]2)=O)C2(CCCCCC2)C1 C1(CCNC(CNS(N)(=O)=O)=O)CN(C(C23CCCC2C3(F)F)=O)CCCO1 CC1C(=O)NCCCN1C(c1cc(CNC(=O)CC2CCC(C)(C)O2)no1)=O C12(C(=O)NCCn3ccc(C(NOCCCC=C)=O)c3)CCC(CC1)C2 Cc1cccc2[nH]c(C(=O)NC3CC3CNC(=O)C=Cc3cccnc3)cc12 C1(C(C)(C)C)CNC(=O)C(=O)N1.C=C1CC1C(=O)NCC C1(C(N(CCCO)CC#C)=O)CCC2CCC1N2C(C1CCCN1CC)=O CCCCC(C)C(=O)NCc1nnn(C)c1C(=O)NCC1CCCN1C(C)=O N1(C(c2c(CCC)nns2)=O)CCCC(C)C1CCNC(=O)CC=CC(C)(C)C C1(=O)C(C)(C)C2=CCN(C2)C(=O)N1CC1(CCN=[N+]=[N-])CC1.c1(COC)c[nH]nc1C C(CCCC(C)NC(c1ccc(-c2cccs2)cc1)=O)NC(C(CC)SC)=O c1(Nc2cc(OC)n[nH]2)cc(N2CC(OC)C(OC)C2)nc(C2CC2)n1 C1(C(N2CC(C)C(CNC(=O)CCS(N)(=O)=O)C2)=O)CCC(C2CCCO2)O1 c1(CNC2CC(C(=O)NC3CC3(F)F)C2)cc(Cl)cc(Cl)c1O c1(C(=O)NC(c2cn(C3CCOCC3)nn2)C)ccc2c(=O)ccoc2c1 c1(C(N2CCN(C(c3cnc(C)s3)=O)CC2CC#N)=O)ccn2ccnc2c1 N1(C(CCc2scc(C#N)c2)=O)CCCC(NC(C2(O)CCCCCC2)=O)CC1 c1(CN(CC)Cc2oc(C)nc2C=Cc2ccccc2)ccc(C#N)c([N+](=O)[O-])c1 C1(C(=O)NCC2CC(C(=O)OC)C2)CCCC(CNc2nn(C)cc2Cl)CC1 N1(C(C(C)CC(F)F)=O)CC2(CC(C(=O)NCC3(CO)CCC3)CO2)C1 C1(SCC(=O)NCC(CC)(C)NC(c2cn[nH]c2)=O)Cc2ccccc2O1 C1(CNC(C(CC)N(C)C)=O)CCCCN1C(=O)CNC(=O)OC(C)(C)C c1(C(=O)NCC(CC(C)C)NC(C(CCC)CC)=O)c[nH]c2ccncc2c1=O N1(C(C(CC)C)=O)CCC(C)CC1CNC(=O)C=CC=C(Cl)Cl C1(NC(C(C)(C)C2CCCCC2)=O)CN(C(C23CCC(CC2)C3)=O)CC1F CCC(CC(=O)NC1CC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C1)C1CC1 n1(CCC)nc(C)cc1C(N1CCCC1CN(C)C(C1CCCC1C(=O)O)=O)=O c1(C(C(=O)NCC(=C)C)N(C)CCNC(C)=O)nc(Cl)cs1 c1(NC(C2C(C(=O)NCCCN3C(C)CCCC3)C2)=O)ccc(Cl)c(C#N)c1 C#CC1(C(N2CC3CCC3(C)C2)=O)CCN(C(=O)CCc2ccncc2)CC1 C1(CNC(C2C(OC)CCCC2)=O)CCC(F)(CNC(=O)CCC2CC2)CC1 c1(C(N2CC(F)(C(C)C)C2)=O)cccc(CNC(=O)CCCn2cccn2)n1 c1(NC(C(c2ccccn2)C)=O)ccc2c(c1)OCC(=O)N2 C=CCC(CC(=O)NCC1CCCCS1)NC(C12CC(C)(CCO1)C2)=O C(=O)(N=c1[nH]nc(C(=O)OC(C)(C)C)s1)NC1CC(c2n(C)cnn2)C1 N1(C(c2c(CC)noc2)=O)CCC2(CCOCC2)C(NC(=O)C(C)CC(N)=O)C1 C1(CNC(C2(OC)CCC2)=O)CCCN1C(=O)C(C)CC1CCCCC1 Cc1ccc(CC(N2CCCC2CNC(C2CC23CCC3)=O)=O)cc1[N+](=O)[O-] c1(CC(c2n(CCC)nnn2)(C)NC(C)CCc2cnccn2)ccc(Br)cc1 c1(OCC)ccc(C(=O)NC(C)C(C)NC(=O)C=CC2CCCC2)cc1Cl C(=O)(CC(CC)C(=O)OC)N1CCC(C(C(=O)NCC2(OCC)CCC2)C)CC1 C1(C(=O)NC2CCCN(C(C(C)n3cnnn3)=O)C2)CCn2cnnc2C1 N1(CCC)CC(n2nc(-c3ccoc3)nc2-c2nc(C)n(CCC#N)n2)CC1=O C1(C(N2CCC(N(C(C3CCC3C(C)(C)C)=O)CC)CC2)=O)CCOCC1(C)C N1(C(C2C(OCC)C2)=O)CCc2c(c(CNC(c3coc(CO)c3)=O)nn2C)C1 C(=O)(C(N=[N+]=[N-])C(C)C)N1CC(N(C(C(C(=O)OC)OC)=O)C)C1 c1(OC)cc(CCC(=O)NCCC(C)NC(C2(C(C)(F)F)CCC2)=O)ccc1Cl C(CNC(c1cc(C2CCC2)nn1C)=O)(C(C)C(C)C)NC(CSC)=O C(c1cn(C(C)(C)CC(=O)NCc2ccccc2)nn1)=C(C)C c1(C(=O)OC(C(C)=O)C)cc(F)c(C)c(N)c1F C1(Nc2nccc(C(=O)OC)n2)CN(C(C2CCC(=O)N2C(C)C)=O)CC12CC2 Cc1cccc2oc(C(=O)NC(C3CCN(C(C4(C)CNC(=O)C4)=O)C3)C)cc12 N1(C(C(C=C=C)C)=O)CCCCC(NC(C2(c3cc(Cl)ccc3F)CC2)=O)CC1 c1(C(=O)NC(=O)Nc2cc(CC)c(C(=O)OC)s2)cccc2cccnc12 c1(C(N2CC(OC)(CNC(C3(C4CCCO4)CC3)=O)C2)=O)cc(C)ccc1C Cc1c(C(=O)NCC(CNC(=O)C(C)c2cnc[nH]2)CO)cnn1CCC(C)C C1(CC(=O)NCCC(COC)(C)O)CN(C(C2(N(C)C)CC2)=O)CC12CC2 N1(C(c2c(C)nsc2N)=O)CCCC(F)(CNC(=O)C(F)CC2CCC2)C1 C1(CC(N2CCC(OCCC)C2)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1C c1(NC(c2c(C(=O)OCC)cccc2F)=O)ccc2c(c1)C(=O)OC2(C)C N1(C(c2c(N)cncc2)=O)CC2CC(C1)N2C(=O)C1=CCOCC1 c1(C(=O)NC2C(O)CCN(C(C3CC(C)C3)=O)C2)cc2c(F)cc(F)cc2[nH]1 C(=O)(C1=CC2CCCC12)NCCCNC(c1c(OC)nccc1)=O CN1CC2OCCN(C(C3CC(NC(C4SC5C=CC4C5)=O)C3)=O)C2C1 C1(NC(c2nc(C)nc(O)c2)=O)CC2CC(NC(=O)CC3CC4(CC4)CO3)C2CC1 C1(O)(CCN(C(=O)C2=CCC2)c2ccccc2)CCN(C(=O)C(=O)NC)C1 C1(C(=O)NCC(N(C(c2cccc(C)n2)=O)C)C2CC2)CC2(CCCCC2)C1 CS(=O)CCC(O)C(=O)NC1(CNC(=O)C=Cc2ccccc2)CCCCCC1 c1(NC(c2ccc(C3(NCc4ncco4)CCC3)cc2)=O)cc(F)c(Cl)nc1Cl C(=O)(NNC(=O)C(C)(C)O)c1ccc(NC(=O)OC(C)(C)C)cc1Cl C(=O)(CCCC(=O)NC1CC(CNC(=O)COc2cnn(C)c2)C1(C)C)OC CCC(C(=O)NCC(C(C)C)NC(=O)Cc1nc[nH]n1)C1CCOCC1 C1(C)(C(=O)NCC2(C)CCN(C(=O)CCCCC3CC3)C2)CC(C2CC2)=NO1 c1(CNC2CCC(C(=O)Nc3ccc(C(C)=O)c(Br)c3)C2)c(O)ccc(F)c1F c1(NCCCN(C(c2n(COC)ncc2)=O)C)nc(C)nc2sccc12 C12(C(N(C(C)CN(C)C)C)=O)CCC(NC(=O)CN3CCSCC3)(CC1)C2 c1(C(N2CCC(NC(c3c(C)cnnc3)=O)C2)=O)csc2c1CCC(C)C2 c1(C(=O)NC2CCCN(C(c3n(C(C)(C)C)ncc3)=O)C2)cnc(O)c(Br)c1 CC1(C)CC(C(N2CC(C3CCCCO3)C2)=O)CCN1Cc1c[nH]c2ncccc12 c1(C(=O)Nc2cc(C)c(NC(=O)Cc3ccoc3)cc2)cc2nc[nH]c2cc1N C1(NC(C(CC)(CC)CC)=O)CN(C(c2cc(C)on2)=O)CC2(CCOCC2)C1 N1(C(CC(c2ccc(O)cc2)C)=O)CCC(NC(=O)CN(C)C2CC2)C(C)(C)C1 c1(CC)cc(C(=O)NCC(CCCC)NC(=O)C=CC(F)(F)F)cc(F)c1 c1(C(N(C(C(=O)NC(c2nncs2)C)(C)C2CC2)C)=O)ncc(F)cn1 c1(C(=O)NC(C(C)NC(CCC#C)=O)CO)ccc2c(n1)NCC2 Cc1cc(F)c(C(N2CC3CC2CCN3C(=O)Cc2nocc2C)=O)c(F)c1 C(=O)(N=c1cc(OC)n(C)[nH]1)C1C(CC)CN(C(C2CCCN2C(C)=O)=O)C1 C1(CNC(C(C)OCCCC)=O)CCCC(NC(=O)C=CC2(C)COC2)C1 N1(C(COCC(C)C)=O)CC(F)(F)CC1CCNC(=O)CC(O)CN(C)C c1(CCC(=O)NCC(C)NC(C2CCc3ccnn3C2)=O)ccc(F)c(F)c1F N1(C(C(C)C#N)=O)CCC(F)(F)C(NC(=O)COc2cccc(F)n2)C1 C#Cc1ccc(C(N2CC(NC(c3csc(=N)[nH]3)=O)C(CC3CC3)C2)=O)cc1 CC1CN(C(C2CC(N(C)C)C2)=O)CC(C)CN1C(=O)COc1ccc(F)c(F)c1 S(=O)(=O)(c1cc(C(=O)NC(C)C(C)NC(c2ccc(SC)o2)=O)co1)NC c1(C(=O)NCCCN2CCN(C(c3cnc(C)o3)=O)CC2)cc(Cl)nnc1O CC1CCN(C(=O)Cn2cnc(=N)[nH]2)CC1C(=O)Nc1cccc(Cl)c1 C(=O)(C(Cc1ccccc1C)CC)NC1(CCCC(C)NC(C(C)SC)=O)CC1 c1(C(=O)NCCC2CCCN(C(C(C)(C)O)=O)C2)c(Cl)cccc1Br C=CC(C)(C)CC(=O)NCCN1CCCN(C(c2cscc2OC)=O)CC1 c1(C(=O)OCCOC2CC=CCC2)cccc(OC(F)(F)F)c1.CC1CNC1=O c1(CC)ccccc1C(N1CCOC(C(C)NC(=O)C(C)N2CCC2)C1)=O N1(C(C(C=C)OC)=O)CCCC(CC(=O)N(c2occc2C)CC2CCCC2)C1 CC1(C)CN(C(=O)CC2CCC(=O)NC2)CC1CNC(=O)C(=O)NC1CC1 N1(C(C(C=C)(C)O)=O)CCCOC(CNC(c2ccc(Br)c(O)n2)=O)C1 N1(C(c2c(COC)nn[nH]2)=O)CCC(CNC(C2CCC(C)(C)OC2)=O)C12CC2 N1(C(C(C)NC(CC)=O)=O)CCCC2(CC(NC(=O)CCC3CCOC3)C2)C1 N1(C(c2cc(CC)on2)=O)C2CCC1CC(NC(=O)C(=Cc1cccn1C)F)C2 c1(CNC(C2(CC#C)CC2)=O)cccc(C(=O)NCc2cncn2C)n1 CCC(CC)C(C)C(=O)N1CCCC(C(=O)NCc2cnn(CCF)c2)C1 CC1(C)C2CCC1(C(=O)NC1CN(C(c3conc3C3CCC3)=O)CC1F)C2 N1(C(C2(CC)CC2C)=O)CC2(CCN(C(C)=O)CC2)c2cc(F)c(Br)cc21 N#Cc1cc(CNC(=O)NC23CC4CC2C3C4)ccc1N1CCCC1 c1(CSC)ccccc1C(=O)NC1COCCC1NC(c1cccc(SC)c1)=O CC1(C)CC(c2cn(-c3c(F)cccc3F)nn2)CN(C(=O)C(O)C(C)(C)C)C1 C1(CNC(C(C)O)=O)CC(O)(CNC(=O)CCN2CCOCC2)C1 CC1CCN(C(=O)CSC2CCCCO2)C(C(N2CC(C(N)=O)C2)=O)C1 C1(CNC(=O)COCC(F)F)CC2(CC2)CN1C(c1ccc(C(F)F)cn1)=O C1(C(=O)NC(C(C)F)C)(NC(C2C3(CC3)C23CC3)=O)CCC(C)(C)C1 C1(=O)CC(C)(C)N1.C1(C(=O)OC)CCN(CC(F)(F)F)CC1 C(=O)(CCCCCNC(C1CCCC(=O)C1)=O)NC(CC#C)C(N)=O c1(CN(C(CC2(OC)CC2)=O)Cc2ccccc2)ccccc1C c1(CNC(C(n2cc(C3CCC3)nn2)C)=O)cccc(OC(F)F)n1 N12CCC(CC1)NC(=O)NCC(C)C2=O.C(CCCN)OCCCCl Cc1cc(CC(=O)NCC2CCC2NC(c2ncncc2F)=O)cc(F)c1 N1(C(C(CCCNC(CNC(C2C(C)C2)=O)=O)O)=O)CCCC2(CC(O)C2)C1 C1(C(N2CC(CC)C2)=O)CCN(C(=O)C(C)(C)O)CCO1 C(=O)(C1=CC2C=CC1C2)N1CCCCC(N(C(C(CCCC)C)=O)C)C1 N1(C(C2N(C)CCC2)=O)CC2CC1CN2C(=O)C(c1cccnc1)O CCCCCC(O)CC(=O)NC(C)CCCC(=O)NCC=CCl N1(C(C(C=C)O)=O)CCCCC2(C1)CN(C(c1cnc(C3CC3)s1)=O)C2 Cc1oc(CNC(=O)C(F)C2CCOC2)nc1C(N1CCCC(C(N)=O)C1)=O c1(CC)c(C(=O)NCC2(C)CCN(C(=O)CC3CCCN3CC)C2)nnn1CC N#Cc1ccc(F)c(NC(C2CCCC(NC(c3ccnc(Cl)c3)=O)C2)=O)c1 C(=O)(C1CN(C(N(C)CCO)=O)Cc2ccccc21)OC(C)(C)C.C1CNC1=O N12CCC(C1)OC(=O)CC1CN(C1)C(=O)C2.c1(CC(=O)NC(C)(C)C)cc[nH]c1 C(=O)(C1=CCC2CCC1N2C(=O)COC)N(CC)CC1CCC1.C(COC)S C1(C)(C(=O)NCC(C)(C)CNC(=O)C(CO)NC(c2ccco2)=O)CC2CC2C1 C1(CNC(c2cn(C)nc2C2CC2)=O)CC2CCC1N(C(=O)CC1CCCO1)C2 C1(CNC(CNC(CN(C)C)=O)=O)CCN(C(C2CC2Cl)=O)C12CC2 CC1(C)CCN(C(C2CC3(CCC3=O)C2)=O)C1C(=O)NCc1cnn(CCF)c1 C(C1=NOC2CN(C(=O)CC3CC(SC)C3)CC12)NC(c1cc(CC)c(C)s1)=O c1(OC)cc(CNC(=O)NC(COC)CO)c(F)cc1Br C1(=CC(=O)NC(C(C)NC(c2coc(N(C)C)n2)=O)CO)CCCCC1(C)C N1(C(C2(n3cc(CCCCCCC)nn3)CC2)=O)CC(CC)OCC1(C)C c1(C(N2C(CC)C(NC(=O)COC3(C)CCC3)CC2)=O)ccc(F)c(C2CC2)c1 c1(C(=O)NC2(C(=O)NCC(COC)OC)CCCO2)cn2c(n1)CCC2 C1(C(=O)NCCC(C)N(C(c2ccc(CC)[nH]2)=O)C)CCOC(C)(C)C1 C1(COC)CN(C(c2cccc(Br)c2Cl)=O)CCN1C(c1c(Br)cccc1Br)=O C=CCCCCCC(=O)N(CCC(=O)N1CC(c2ccccc2)C1)C(C)C N1(C(COCCCC)=O)CCCC(C)C1CCNC(=O)CC(F)(F)F C1(CC)CC(CNC(c2ccc(Br)cc2)CO)CCO1 Cc1cc(NCC2C3CN(C(C4(O)CCC(C)CC4)=O)CC23)ncc1[N+](=O)[O-] C12(OC)CCCCC(C(N3CC(NC(c4ccc(C)cc4N)=O)C3)=O)(C1)C2 C1(N2C(CNC(CC)=O)(CNC(=O)CC(C)C(C)C)CCC2)CCc2nnnn2C1 C1(CC(=O)NC2CC2NC(c2ccc(C(F)(F)F)c(Cl)c2)=O)CCCC(F)(F)C1 N1(C(C2C=CCN2Cc2ccc(Br)cc2Cl)=O)C2CCC1CC(O)C2 C=CCCCC(=O)NCc1cc(C(N2CCC(C(=O)NCC)C2C)=O)n(C)n1 C12(CC)CN(C(c3cnccc3C)=O)C(CNC(=O)C(F)C3CCOC3)(C1)C2 N1(C(=O)NC(c2ccc(CC)cc2)COC)CCOC2CN(C(C)=O)CC12 c1(C(N(CCC)CC2CCOC2)=O)cc(S(=O)(=O)N2CCSCC2)c[nH]1 C1(CCNC(C(C)N(C(=O)Cc2ccsn2)CCC)=O)CC(=O)N(C)C1 O=C(C1=CS(=O)(=O)CCC1)NCC1CCC1NC(c1cc2sccc2cn1)=O Cc1ccnc2sc(C(=O)NCC(C)NC(=O)C(F)(F)C(O)C(C)C)c(C)c12 Cc1cc(N)ccc1C(N1CCCC1C1CCCN(C(=O)Cc2cnoc2)C1)=O c1(C(N2CCC(C(C)NC(=O)CN3CC(C)(C)C3)C2)=O)nnn2c1CCCCC2 N1(C(CC(OCC)OCC)=O)CCC(O)(C(=O)NC2CCC(CC)CC2)CC1 CCCC(F)C(=O)NCCC(CNC(C1CC(C)(CC)C1)=O)OC CCCC(C)(CCC)NC(C)C(c1ccc(F)c(F)c1)O c1(C(=O)NCC23C(CN(C(C(CC)C#N)=O)C2)CC3)cc(Cl)c(Cl)cc1Cl C1(C(=O)NCc2occ(C(=O)NC3(C(C)(C)C)CCCC3)n2)CCC=CCC1 c1(OC)ncc(C(=O)NCC(C2CCCN2C(=O)CSC(C)C)(C)C)cc1Br c1(OC)cccnc1CC(N1CCSCC1C(=O)O)=O N1(C(C=C(CCC)C)=O)CC2C(CN(C)C(c3ncn(C)n3)=O)C2C1 c1(C(C(=O)Nc2c(C)cccc2C)N(CC=C)C(C)C)cc(C(F)F)cc(C)c1 C(C)(CCCCNC(c1csc(COC)c1)=O)NC(c1n(CC)ccc1)=O C(N=c1[nH]c2c(c(=NCCCC(C)CO)[nH]1)CCC2)c1c(C)nc(CC)n1C c1(OC(C)C)ccc(NC(=O)CC(N)C(F)F)c(I)c1 C(C)(CCC(=O)N1CCCC1C(=O)NC(C)CC(C)C)OC c1(NC(C2CCC(NC(C3CCCN(C)C3)=O)C2)=O)cc2n(n1)CCNC2=O c1(C(N2CCN(C(CCSC)=O)C(CCO)C2)=O)cc2c(cc1F)OCC(=O)N2 c1(CNC(N(CC=C)C)=O)nccc2c(C)cccc12 C1(C(=O)NCc2c(N)non2)(CNC(=O)CC2CCCC(O)C2)CCCCC1 C(c1ccc(C)cc1)=CCC(=O)NC1C(NC(c2c(CC)noc2)=O)CCCC1 c1(CNC(C2CCN2CC2CCC(C(=O)O)CC2)=O)cccc2c1CCCC2 C12(NC(CSCC=C)=O)CCCCCC1N(C(c1nn(C)cc1[N+](=O)[O-])=O)CC2 C1(NC(CC(C)C2CC2)=O)CC2(CCN(C(=O)Cc3ccc(O)nc3)CC2)C1 c1(C(=O)NCC(C)(C)NC(C2C(C(C)C)OCC2)=O)ccnc2ccnn12 C(=O)(CC(=O)NC12CC(NC(=O)C(C)(F)F)(C1)C2)OC c1(C(N(CCCN(C(C2CCC(C)O2)=O)C)C)=O)nn(C)cc1S(N)(=O)=O c1(-c2cn(CC3N(C(C4CC4C(=O)O)=O)CC=C3)nn2)ccc(F)cc1 N1(C(CNC(=O)COc2cn[nH]c2)=O)CC=CCC1.C1COC1 C1(NC(CC)=O)CC2CN(C(c3ncccc3COCCOC)=O)CCN2C1=O c1(C(CNC(C=C(C)CNC(=O)CCCn2ccnc2C)=O)=O)cnc(C)[nH]c1=N CC(C)C1=NOC(C(N2CC3(CC3)CC2C)=O)C1 c1(CNC(C(C)Cn2ccnc2)=O)cccc(NC(=O)Cc2ncc(Cl)s2)c1 Cc1cccc(C(O)C(N2CC(CNC(=O)Cc3cn(C)cn3)C(O)C2)=O)c1F C1(NC(C=C(C)CNC(C2C3C4CCC(C4)C23)=O)=O)CCc2ncnn2C1 N1(C(c2sc(C)c(O)n2)=O)CC2CN(C(c3c[nH]nc3C3CC3)=O)CC2(C)C1 C(=O)(CC(O)CN(C)C)NC(CN(C(c1cn(CC=C)nn1)=O)CC)CC OC1(c2nc(-c3ccco3)no2)CCNCC1 C(CCCCC(=O)NCCC(=O)NOC1CCCCC1)NC(C1N(CC)CC1)=O C(C(C)(C)CC(=O)NC(C)C(=O)NCc1nc(C)c(C)[nH]1)OC(C)=O CC(CCC(=O)NC1(CF)CCN(C(=O)C(C2CC2)C2CC2)C1)N(C)C CC1CN(C(=O)C(CC#N)c2nnc(NC(=O)OC(C)(C)C)o2)CC(C)C1(C)O C=CC1CCN(C(=O)C(CCSC)NC(C2CCC(=C)CC2)=O)C1 C1(O)(C(C(=O)NC2CC(CC(=O)NCCN(CCO)CC)C2)F)CCCC1 C1(CC(=O)NCCC2CC(CNC(CC(=O)NCC)=O)C2)CC(=O)NC1=O c1(C(N(C(C)CCNC(C2CC2C(F)F)=O)C)=O)ccn2nnnc2c1 C(=O)(CC(C(F)(F)F)n1ccnc1)N1CCN(C(=O)Cn2ccnn2)CC1CF c12cccc(c1)S(=O)(=O)N1CC3C(C3C1)NC2.c1(C2(C)CC2)ccc(C(=O)O)s1 C1(C)(CNC(CCCSCC)=O)CN(C(=O)OCCNCC2CCO2)C(C)(C)C1 CC(C)C(C)(F)CNC(=O)COC1CN(C(C2CC23CC3)=O)C1 c1(CNCc2c(C)n3c(s2)cnc3)ccc(F)c2c1CCC2 C1(NC(C2C(C=C)C2)=O)COCC1CNC(C1(CSC)CCC1)=O C1(C(=O)NC(CCO)C(C)(C)O)(CC)CCCN(C(=O)CCCOC(C)(C)C)C1 C1(COC)CCOCC1.C(=O)(C(CCl)OC)NCCOCCN(C(=O)N)C.OC C(CCCC(=O)NCC1CC(O)(CNC(C2CC2(F)F)=O)C1)N(C)C C(C(C)(C)CNC(=O)COCCN(C)C)C1CN(C(C2C(C)C2)=O)C1 C1(C(N2CC(N(C(C(C)O)=O)C)C2)=O)CCOC(=O)N1 Cn1c(CN2CC3C(NC(=O)Cc4ccc(F)c(F)c4)C3C2)cc2ccccc12 c1(C(N(CCCNC(COCCCNS(CC)(=O)=O)=O)C)=O)cc(C)[nH]n1 N1(C(CCNC(=O)OCC)=O)CC(CC(=O)NCC2C(CO)C2(F)F)CC1(C)C c1(C(=O)NC(CSCC)C(=O)N(C)CC)ccnc(C)n1 C1(C(=O)NCC(CCC)NCc2c(C)n[nH]c2C)CCC(CO)CC1.C1(=O)CO1 CC1(C)COC(C(=O)NCCCN(C(c2csc(Cl)n2)=O)Cc2ccccc2)C1 C(=O)(C1=Cc2ccccc2C1)N1C(CC(N2CC3(CCC3)CC2CO)=O)CCC1 C1(O)(CC(=O)NCC2(C(=O)NC3C(C4C(C)C4)C3)CC2)CCCCCC1 C12C3CCCN(C3C1(C)C)N(C1CC1)C2=O.Cc1nnc(Cn2cc(CN)nn2)o1 N1(C(c2c(OC)cccn2)=O)CCc2sc(C(N3CCC(C)C(F)C3)=O)cc2C1 CCC(C)(C)C(=O)N(C1CCC(NC(c2nc(C(F)(F)F)cn2C)=O)CC1)C C(=O)(C(F)(F)C(O)C(C)C)NC1CCN(C(CCSCCCC)=O)C1 c1(C2C(C(NOCC(CC)C)=O)C2)ccc(C(=O)OC)nn1 N1(C(Cc2nnc(C)o2)=O)CCC(N(C)C(c2cc(CC(C)C)nn2C)=O)C1 N1(C(C(C)F)=O)CCCCC1Cn1cc(-c2cccnc2Br)nn1 CC(Cn1cccn1)C(=O)N1CCC(CCNC(C2CC(C(C)(C)C)C2)=O)C1 N1(C(C2CC(O)C2)=O)CCN(CC2CC=CC2)C(=O)C1 C#CCCCC(C)C(=O)N(CC(=O)NC(CCSC)C(C)C)C c1(C(=O)NCC(C)NCc2nc(C)c(COC)s2)cccc2cc[nH]c12 CC1CN2CCN1C(C(=O)NC(CNC(C1(C3CCCCO3)CC1)=O)C1CC1)C2 C#CCCCCC(=O)NCCN(C1CCCC1)C(C1CCN(CC(F)(F)F)C1)=O C1(NC(c2ccc(C(C)O)cc2)=O)CN(C(c2coc(C3CC3)n2)=O)CC1(C)C C(=O)(C(CC#CC)NC(c1ccncc1Cl)=O)NCCC=CC C1(CC)CCN(C(C)=O)C1C=O.C(=O)(C(C)(C)C)NCCOCCF N1(C(c2nnn(C(C)(C)C)n2)=O)CCCCCC1CNC(c1coc(Cl)c1)=O N1(C(c2cc(C)no2)=O)CCCC(C)C1CNC(=O)C(c1ccc(F)cc1)(C)F C1(C)(C(=O)NC2CN(C(c3ccc(C)nn3)=O)CC2C)CCCCNC1=O N1(C(CC(C=C)C)=O)CCCN(C(c2cccc(Cl)c2COC)=O)CC1C n1(CC(=O)NCC(C)(C)F)cc(CNC(=O)CCOCC(F)F)nn1 C12(C(=O)NCC(C)(CNC(C3(C)CCCCC3C)=O)OC)CC3CC1C2C3(F)F c1(C(N2CCN(C(Cc3cccc(C)c3)=O)C3C2C3)=O)cnc2nccn2c1 C(=O)(C1CCCc2c1ncn2C)NCC1C(F)(F)CCN(C(C(=O)N(C)C)=O)C1 CCCC(C(=O)NCC=C1CCN(C(c2nn(C)cc2N)=O)CC1)NC(N)=O C1(NC(COCCC=C)=O)CCCC12CCN(C(C1CCCC(C)C1)=O)CC2 c1(C(N2CCN(c3cccc(C)c3)CC2)=O)ncc2n1CCCC2 N1(C(C(C)O)=O)CCC2(CCC(CN3C(=O)NC(C)C3=O)O2)CC1 c1(CC(=O)NC(C2CCCC2)CN(C(CC(=C)C)=O)CC)ccc(F)c(Cl)c1 C1(C(=O)NC2(CC=C)CN(C(C3CCCCN3C(C)=O)=O)C2)CC(C(C)C)=NO1 CC(C)(C)CC(O)CC(=O)NCC1CCN1C(c1ccc(Cl)cc1OC(F)F)=O c1(CC)ccc(NC(=O)CC2CCCC2NC(c2cnc(C3CC3)o2)=O)cn1 N1(C(C)=O)CSCC1C(=O)NCC1(C)CCC1.C12(CCC1)CCN(C(C)C)C2=O C(CCN(C)C(C1(C)CC2CCC(C1)S2)=O)(C(C)(C)C)NC(C1CC(OC)C1)=O c1(C(N(C(C)C(=O)NCC2CCC(=O)O2)CCC)=O)ccc(F)c(O)c1 N1(c2snc(C)c2C#N)CCC12CCCOC2 n1(CC(=O)NC2C3CN(C(C4C(C=C)C4)=O)CC2C3)nc(C(F)F)c2c1CCC2 c1(C(N2CCCC(CO)(NC(C3CC(O)C3)=O)C2)=O)ccn2nccc2n1 c1(C(N2CCC(C(=O)NCC(CC)(CC)CO)O2)=O)nccc2[nH]ccc12 CC(C)C(O)C(C)C(=O)NC1(CNC(=O)C2=COCCC2)CCCCC1 CC(C)C(C(=O)N1CC(CN(C)C(C2CCCC23CC3)=O)C1)C1CCCCC1 N1(C(CC(C(C)C)OCC)=O)CCC2OCCN(C(c3ccc(CC)s3)=O)C2C1 C12(CNC(C3N(CC)CCC3)=O)CCC(CC1)N2C(c1cc(N)c(F)cn1)=O Cc1ccc(CC(=O)NC2CC(C(C)NC(=O)C(C)c3ccsc3)C2)cc1C C(CC1=CCN(C(=O)CC(C)n2ccnc2)CC1)NC(C1C(OC)(OC)CC1)=O c1(C(N(CCCCCNC(=O)Cc2cnc[nH]2)C)=O)cc2ccccc2cc1Cl C1(NC(C2(OC)CC2)=O)CCCCN(C(C2CN(C)CCO2)=O)C1 C1(C(=O)NC2(C)CN(C(C3C(CN(C)C)C3)=O)C2)C(F)(F)C12CCC2 CC1CN(C(c2c[nH]nc2C(C)(C)C)=O)CC(C)N(C(=O)C2=CCC2)C1 C(c1nc2ccccc2s1)=CC(=O)N(C1CC1)CC1N(C(C(C(C)C)F)=O)CCC1 CN1CCC(C)(C(N2CC=C(CNC(C3CC4CCCCC34)=O)CC2)=O)C1=O N1(C(C2CC3C=CC2C3)=O)CCC2C1CCCN2C(c1ccc(Cl)c(F)c1)=O c1(CC(N2CCC(CCNC(=O)C=Cc3cscn3)C2)=O)ccccc1C1CC1 C1(CN(C(C2(C#C)CC2)=O)C)CN(C(c2c[nH]c(=N)s2)=O)CC12CC2 c1(C(=O)NC2CN(C(c3c(C)cc(C)nc3)=O)CC23CC3)ccc2cc[nH]c2c1 C1(CC(=O)NC2(n3cccn3)CC2)CCCCC1(C)C.C12CC(C1)C(=O)NC2C CC(C)C(C)CN(CCC(=O)NCCCN(C(c1coc(Br)c1)=O)C(C)C)C CC1(NC(=O)CCc2ccncc2)CCCCC1C(=O)NCC1CC1c1ccco1 C(=O)(C1=CC2(CCOC2)C1)NCCN(C(c1cnc(CC)nc1C)=O)CC C#Cc1ccc(CC(=O)N(C2CN(C(=O)C3CC3)CC2(C)C)C)cc1 N1(C(C(C=C)(C)O)=O)C2CCC1CC(CNC(=O)CC1CCOC(C(C)C)C1)C2 C1(CNC(CCCOC(C)=O)=O)CCCCC1NC(=O)CN1CCC(C)CC1 C1(CNC(CCOCCCOC)=O)CCN(C(c2ccc(F)nc2F)=O)C1(C)C c1(CCC(=O)NCC(C)(C)CNC(=O)C(=O)NC2CC2)ccc(Br)cc1 c1(C(=O)NC2CCC(CCNC(C3(CCOC)CCC3)=O)C2)cc2occc2[nH]1 C1(CNC(=O)CO)CCN(C(C2CC(OC(F)F)C2)=O)CC1 c1(N2CC(COC(C3CC(C)C3)=O)C2)ccc([N+](=O)[O-])c(Sc2ccccc2)c1 N1(C(CC2CCCC(C)O2)=O)CCC(C)(C)C1C(=O)NOCC(F)(F)F c1(OC(c2cncc(OCC)c2)=O)ccc(F)cc1CCOC c1(C(=O)NCCC(O)CNC(C2CC2CF)=O)ccc(OCC(F)(F)F)nc1 Cc1ccnc(Cl)c1C(=O)NC1CCC(NC(=O)CCc2cc(Br)ccc2F)C1 c1(C(=O)NCC2(C(C)NC(=O)Cn3cnnn3)CC2)cc(O)nc2c1CCCC2 C1(C)(CNC(C(C)CN(C)C)=O)CCC(NC(=O)Cn2ccc(C3CC3)n2)CC1 CCC(CC)C(=O)NC1C=CC(CC(=O)NC2(C(N)=O)CCCCC2)C1 c1(-c2[nH]nc(C(C)C)n2)ccc2c(c1)OCCO2 C1(NC(c2c(C)scc2)=O)CN(C(=O)CCOCC2CC2)CCC12CCC2 C(C(O)C(C)c1ccccc1)NCCCN(C(C(C)N(C(=O)OC)CC)=O)C1CC1 N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(c2ccc(C(=O)NC)cc2)=O)CCC1C c1(CN2CCC(NC(CC(CC)CN(C)C)=O)CC2C)nc2ccccc2o1 c1(C(=O)NCC23CC2CN(C(=O)CC2(CO)CC2)C3)ccc(Cl)cc1O C1(NC(c2c(CC)ocn2)=O)(CC)CCCN(C(c2cncc(OC)n2)=O)C1 c1(C(=O)NC2CN(C(CCc3ncc(C)[nH]3)=O)CC23CC3)c[nH]c2ccccc12 C(=O)(C1SCc2cccnc21)N1CC(C)N(C(c2cccc(=O)o2)=O)CCC1 c1(C(=O)NCC(CC)NC(c2ccc(C3CC3)nc2C)=O)noc2c1COCC2 c1(C(N(C(c2ccccc2)CNC(CNC(CCC)=O)=O)C)=O)cc(C#N)no1 C1(NC(C2CC(CC)C2)=O)CCCC(NC(c2ccccc2OC(F)F)=O)C1 c1(CCOCC(=O)N(C2CCN(C(C3COCCO3)=O)C2)C)ccccc1 C#CCC(C)(CNC(=O)C(O)CCCNC(=O)C(CO)OC)CO N(C(=NCCCF)N1CCC(OC)C(C)(C)C1)CC1(CC)CCC(=O)N1 CCCC(CC)C(C(=O)NCC1CCCC1)N1CCCC(Cn2ccnn2)C1 c1(C2C(C(=O)NCCC(C)NC(=O)C=Cc3cocn3)C2)cnn(C)c1 c1(OC(C)C)ccc2c(c1)C(NC(=O)C(=O)NC1CCC1CN)CCO2 C1(NC(c2n(CC)nc(C3CC3)c2)=O)CN(C(=O)CC(C)OC)CC1C1CC1 CCC(CC(=O)NCc1nn[nH]n1)NC(c1cn(C)nc1C)=O C(CCCC(C)C)NC(C(CN(C(CC(C)OCCCC)=O)C)C)=O c1(SNCC(=O)OC)ccccc1NC(=O)N(C(C)CCC(C)C)C c1(C(=O)NC2C3(CC(NC(C)=O)C3)C2)ccc(C)nc1Cl N1(C(CCC(C)SC)=O)CCCC2C1CCN2C(=O)C=CCN1CCCC1 N1(C(C(C)NC=O)=O)CC(C)(C)CC1CC(=O)NCCCc1ncn(C)n1 c1(C(=O)OCC(c2c(OC)cccc2)=O)ccc(F)c(OC)c1F C1(OC)CN(c2cccnc2)CC(C)(C)C1.C12CC3CN(CC13)C2=O c1(C(N2CC(CC(=O)NCCCc3cn[nH]c3)OCC2)=O)cc2n(n1)CCCC2 C(=O)(C(C1CC1)N(C(=O)C(F)C1CCCC1)C)NCCSCCOC N1(C(C(C)Cn2ccnc2)=O)CC2(CC(CC(=O)N(CCCN)C)C2)C1 c1(NC(C2OCCN(C(c3nc(C)oc3)=O)C2)=O)ccc2nnsc2c1 c1(C(=O)NC2C(F)(F)CCN(C(C3CCN(C)C3)=O)C2)cc2cccc(F)c2s1 C1(NC(=O)CNC(=O)C2CC2)CC(F)CN(C(=O)C=Cc2ccccc2)C1 CCC(CC)CCC(=O)NCCN1CCN(C(c2cnnn2CC)=O)CC1 CCCCCCC(C)C(=O)N1CC2CC1(C(N1CCCC1C1CCOC1)=O)C2 c1(CC(=O)NCCCN(CCCNC(C2(C)COC2)=O)C)ccc(O)nc1 C(=O)(CCCC(=O)NC(c1ccc(F)cc1F)CNC(C1CC1(Cl)Cl)=O)OCC c1(Cn2cc(CC3N(C(n4cc(CO)nn4)=O)CCC3)nn2)ccc(F)cc1 C12(NC3(C)N(C)CC(OC)C3)CCCN(CC1)C2 C(CCCCC(=O)NCCC1CCC(C)C1)N(C(C(C)=CC(C)(C)C)=O)C CCCCC(CC)CCC(Cn1c(NC)nnc1-c1csc(CCO)n1)CC C(C)(CO)(C(=O)NCCCCCF)NC(c1cc(C(C)C)no1)=O c1(C(N(C2(CC(=O)N(C(C)CS(C)=O)C)CC2)C)=O)ncccc1O C1(NC(c2cncc(C#C)c2)=O)CCN(C(C2COC3(CO)CC2C3)=O)CC1(C)C N1(C(c2cc(C)n(C)n2)=O)CC2(CCOCC2C(=O)NCc2cnccn2)C1 c1(C(=O)NCC(C)NC(=O)C=Cc2ccncn2)cc(N)cc(O)c1 C1(NC(CSC)=O)CN(C(=O)C2CCOc3ccccc32)C2(CCOCC2)C1 C1(CC(=O)NCCN(C(c2csc(C(F)F)n2)=O)CC)CC2(CCOCC2)CO1 N1(C(CCC(C)C)=O)CCCC2CN(C(c3cc4c(s3)CC(C)CC4C)=O)CC12 C1(CCC(=O)N(CCCCO)C2CC2)CCCCN1C(c1ccccn1)=O c1(C(N2CCOCC(NC(C(C)n3ccnc3)=O)C2)=O)c([N+](=O)[O-])cnn1C C1(O)(CNC(C2(C(C)NC(C3CCSC3)=O)CC2)=O)CCN(C)CC1 c1(NCC2(CNC(C3CCC(C)(CC)O3)=O)CC2)nnc(C)c(C)c1C#N c1(C(N2C(C(=O)Nc3cccc(F)c3)CCC2)=O)ccc(CO)cc1 C(c1cccc(O)c1)=CC(N1CCC(C)(C(=O)NC2(CO)CC2)C1)=O N1(C(c2c(C#N)scc2)=O)CC2CC(C1)N(C(C1CC3(CSC3)C1)=O)C2 N1(C(Cc2c(C)ccs2)=O)CCOCC(CNC(=O)CCCC2CCCC2)C1 CC1(C)CCC(NC(C2C3CCC(C3)N2C(c2cccc(C(N)=O)c2)=O)=O)CC1 N1(C(CSc2n(C(C)C)cnn2)=O)CC2CC2(CNC(=O)COC(F)(F)F)C1 C#CCCCC(C)C(=O)N1CCC2CC12C(N1CCC(C)C(O)C1)=O CC1CN(C(c2cnc(C3CC3)o2)=O)CC1CCNC(C1CS(=O)C1)=O C1(NC(c2cc(CC)on2)=O)CN(C(c2cccc(OCCO)c2)=O)CC1F C(=O)(CCC(=O)N1CC2CC1C2NC(=O)CC1(C)CC1)c1ccc(C)s1 O=C(N=c1c(Br)c[nH]cc1I)C1CC(NC(=O)CCc2ncc[nH]2)C1 c1(C(N2CC3(C(NC(=O)C=CC4CCCO4)CC3)C2)=O)cccc(Cl)c1[N+](=O)[O-] C1(OC(=O)CNC(=O)C2CC2)CCCC1CNC(C1(C2CCCO2)CCC1)=O N1(C(c2c(NC)snc2C)=O)CCC2(CCC2)C(NC(=O)C(C)=C2CCC2)C1 c1(C(=O)OCC2C(c3n(C)ncc3)C2)c(Cl)ccnc1F c1(NC(=O)OC(C)(C)C)c(C(=O)NCCCCCSCC)cccc1C C1(C(N2CCC(CCNC(C3(C)CC=CC3)=O)CC2)=O)CSC2(C)CCC(=O)N12 CC(C)CC(O)CNC(c1cccnc1)Cc1cccc(Cl)c1 Cc1nc(C2CC2)oc1CNC(C1CC1)=O.c1(OC(C)C)nccnc1O C1(CC(C)NC(C2CCCN2C)=O)CCN(C(C2(C(F)(F)F)CCCC2)=O)CC1 Cn1nccc1C1(NC2C(NC(=O)C(N)=O)CCC2)COC1 c1(C(N2CC3C(N(C(=O)Cc4ccc(F)cn4)C)C3C2)=O)cc(F)c(F)cc1N CC1(C)CCC2(CC1)CC2C(N1CC(NC(c2cc(Cl)ccc2N)=O)C1)=O C1(C(=O)NCc2cnn[nH]2)CCCN1C(=O)C(F)OC(F)(F)F c1(C(=O)NCCN(C)C(c2cc3n(c2)CCC3)=O)ccc(OC(F)(F)F)cc1Cl c1(C2N(C(C(C)O)=O)CCC2)ccc2c(c1)CCO2 N1(C(CCC(N)=O)=O)CCCC(F)(F)C1.C12CC1C(=O)N2 c1(C(=O)OCC)ccc(S(=O)(=O)NC(COC)C2CCC2)o1 C(C)(CNC(=O)CCc1ccc(C)o1)(CNC(c1cscn1)=O)OC N1(C(C(c2ccc(C)s2)C)=O)CCCC(NC(c2c(C)ncnc2O)=O)CCC1 CCCCC(=O)C(=O)NCC12CCC1CN(C(c1ccncc1NC)=O)C2 c1(C(N2CCC(NC(C3C(=C)CC3)=O)(CO)C2)=O)cc(C(C)C)ccc1F N1(C(C2(CC)CCNC2=O)=O)CC(NC(=O)CNC=O)CC2(CCC2)C1 CCC(CC(C)C)C(=O)N1CC(OCCC(=O)NC(C)(C)C(C)(C)C)C1 c1(C(C(=O)NC2CCC2)N(CC(CC)C)Cc2cnn(C)c2)cc(O)nc(O)n1 N1(C(CC2(C=C)CC2)=O)CC(OC)CC(NC(c2cc(COC)nn2C)=O)C1 C1(C(N2CCC(CN(C(CCCN(C)C)=O)C)C2)=O)CC(=O)N(C2CCCC2)C1 CN1CCC(=O)Nc2cc(C(=O)NC3(C)CCOC3)ccc21 N1(C(CN2C(=O)CN(C)CC2)=O)CCC(CF)C1.C(=O)(C(C)C)N.CO C(=O)(CC(C)CCC(=O)N1CCN(C)CC1CNC(C1CS(=O)(=O)C1)=O)OC c1(NC(C2C(NC(c3c(C)nccn3)=O)C=CCC2)=O)cccc2c1OCC2 c1(C(=O)NCC2C(NC(CCn3ncc(C)c3)=O)C2)ccc(-n2ccnn2)cc1 C12CCC3(CC1)CN(CCO3)C(=O)C1(CC1)CNC(=O)CS2.N1(CC)CCCC1.C Cc1nncn1CCNC(=O)CC1CC(NC(=O)CCn2cc(C)cn2)C1 N1(C(CCCOCC=C)=O)CCC2C(C1)CN2C(=O)C(F)C1CC1 Cc1ccc(NC(=O)CN(c2c[nH]c(Br)c2)C)cc1O N1(C(Cc2cccc(OC)c2)=O)CCC(C)(NC(=O)Cc2csc(CO)n2)CC1 c1(C(N(CCCNC(c2c(CC)c[nH]c2)=O)CCCC)=O)ccccc1C(N)=O C12(C(=O)NCC(C(=O)NCC(=O)OC)N(C)C)CC(C#N)(C1)C2 c1(C(=O)NCC(CC(=O)NCC(CCC)(C)O)C2CCC2)ccc(C)c(C)n1 C1(CNC(C2CCC(C)CC2)=O)C2CCCC1N(C(c1csc(=N)[nH]1)=O)C2 Cc1nc(O)nc(O)c1CCC(=O)NC12CC(NC(=O)CC3CC3(C)C)(C1)C2 Cc1cc(C)c(C(=O)NCC(C)(C)NC(C2CCC(C)(C)CC2)=O)cc1Br c1(OC)cc(C)cc(C(N2CC3(CCC(CNC(=O)C=CC(C)C)O3)C2)=O)c1C c1(C(=O)NC(C)CCCCNC(=O)CCC2CCOC2)cnc2ncccc2c1 N1(C(C2(CO)CCN(C(=O)C(c3ccn(C)c3)C)C2)=O)CC=C(CCOC)CC1.CO c1(N(C)CCc2cnccn2)nc(N2CCC(S(C)(=O)=O)C2)c2c(n1)CCS2 c1(C(=O)NCC23N(C(C(CCC#C)O)=O)C(CC2)CC3)cnnc2ccccc12 Cc1ccc(F)c(C(=O)N(C(C)C(=O)NCc2cn(C)cn2)C2CC2)n1 c1(C(=O)OC)cc(OC)c(-c2nnnn2C)cc1OC(C)(C)C N(C(=NCCC1CCCS1)NCc1ccccc1F)CC(C)Oc1cccc(F)c1 C123CC(CN1C(=O)CSC)(C2)CC(C1CC1)C(=O)NC3.C(COCC)OC.OC CC(C#N)CN=C(NCc1ccc(C#N)cc1)NCc1ccc(Br)cc1 Cc1ccc(OC(F)F)c(Cl)c1.N12CCN(CC1)C(=O)C1CN(C1)C(=O)CC2=O c1(OC)cc(C(=O)NCCOCCn2cc(CSCCO)nn2)[nH]n1 C1(CNC(CSCC=C)=O)CCN(C(c2cn(CCCC)nn2)=O)CC1C N1(C(=O)COC2CC=CC2)CC2(C1)CN(C(c1ccc(Cl)nc1Cl)=O)C2 C(CCC(C)CC(C(=O)OCC)N(CC(C)(C)COCC(=O)OC(C)(C)C)C)=CC=C N1(C(c2cc(OC)nc(F)c2)=O)CCN(C(=O)COC(F)(F)F)C(C)CC1C c1(CC(=O)NCC2C(CO)C2(F)F)cn(Cc2ccccc2)cn1 c1(C(=O)NC2CCC2NC(=O)C(O)CC2CCCCC2)csc([N+](=O)[O-])c1 N1(C(c2c(CC)nns2)=O)CCN(C(C2(COC)C=CCC2)=O)CC(O)C1 N1(C(c2cnc3n2CCOC3)=O)CCCC2(CCCN(C(C3CCC3)=O)C2)C1 C1(CC(=O)NCC2CCC(NC(c3nn(CC)c(O)c3)=O)CC2)CCC(C)(C)CO1 c1(OC)coc(C(=O)NCC(C)(O)CNC(C2CC(CC(C)(C)C)C2)=O)cc1=O Cc1cc(CCC(=O)NC2CCCN(Cc3cc(C#N)ccn3)C2)cc(C)n1 C(=O)(CC(C)C(=O)OC)NC(CC)C(=O)N1CCC(SC)C1 C(CCCCCF)NC(C1CC(NC(=O)C(F)n2ccnc2)C1)=O C1(CC(=O)NC2C3CC(CNC(C(CCC)O)=O)(C3)OC2)CCN(OC)CC1 C1(C2CC2)(CC)CN(C(=O)C(CC2CC2)NC(=O)COc2cccnc2)C1 C1(C(=O)OC)CC(C)N1C(=O)CN(C1CN(C(C2CN(C)C2)=O)C1)C Cc1ccc(NC(=O)C(=O)NCC2(O)CCCNC2)c(Cl)c1 N1(C(C(C(C)C)CSCC)=O)CC2CCN(C(c3nc4ccccc4[nH]3)=O)CC2C1 C(=O)(CCC(=O)NCC1COCC1NC(=O)CCc1ccc(CO)cc1)NC Cc1cccc(C(=O)NCC(C)(C)NC(C2CCC(O)C2)=O)c1 c1(C(=O)NC2CN(C(C(C)OCCOCC)=O)CC2C)ccc(F)c(C#N)c1 Cc1ncnc(C)c1C(=O)NC1CC(C)CN(C(C2CC2C(F)F)=O)C1 c1(C(=O)OC)nnn(C2CCN(CC(N3CC(C)C(F)C3)=O)CC2)c1C(F)(F)F C(=O)(C(C(C)C)NC(c1ccc(Cl)cn1)=O)N(CCC(C)NC(CC(=C)C)=O)C c1(C(=O)NCC2CC(NC(c3ccncn3)C)C2)cncc(C(F)F)c1 Cc1nc(C(=O)NCC2(NC(=O)Cn3nnnc3C)CCC2)ccc1C#N C(CCC(O)C(=O)N1CCCCC1C(F)F)NC(c1ccn(COC)n1)=O C1(CNC(CNC=O)=O)CCC12CCN(C(=O)C=Cc1ccc(O)c(O)c1)CC2 c1(NCC2(O)CN(C(c3c(SC)scc3)=O)C2)ncnc2c1ncn2C C(C)(C)(C(C)CC(=O)NCc1cnc(COC)[nH]1)NC(c1n(CC)ccn1)=O c1(C(=O)NC2C(NC(CCc3ccc(C)cc3)=O)CC2)ccc(O)c([N+](=O)[O-])c1 CC1CCC=C1C(=O)N1CCC(NC(c2cc(=O)cc[nH]2)=O)C12CC2 c1(C(C(=O)O)NC(=O)NCc2c(C)ncs2)cnc(O)nc1 N1(C(c2c(C)nc(CC)o2)=O)CCC(C2CC2NC(=O)C(C)(F)CC2CC2)CC1 c1(C(N(CC(C)N(C)C(C2CCCN2N=O)=O)C)=O)cccc(C(C)(C)C)c1 C1(NCc2c(C)nn(CC)c2C)CS(=O)(=O)C12CCOCC2.c12ccccc1C2 n1(CCC(=O)NCC(CNC(C(C)=C(C)C)=O)C)ncn(C)c1=O C1(CNC(C2C(NC(c3cc(OC)no3)=O)CCCC2)=O)CC2CCC1CC2 N(C(=NCc1ccncn1)NC1CCOCC1)CC1CC(F)(F)C1 N1(C(C(n2cc(C)nc2)(C)C)=O)CCC(NC(=O)C=CC2CC2)C(O)C1 CCCN=C(NCc1ccccc1C1CCC1)NCc1ccc(C)cc1 c12cc(ccc1C(C)C)C(=O)N2.C(C(C1CCC1)OCCC)OC [N-]=[N+]=NC1(C(=O)NC2CCC2NC(c2ccc(C(F)(F)F)[nH]2)=O)CC1 c1(NCC)cccc(CN=C(NC(C)C2CC2)NC2CC(=C3CC3)C2)c1 c1(C(=O)NCCC2(NC(Cn3c(C)ccn3)=O)CC2)ccc(-n2ccnc2)nc1 c1(OC)sccc1C(N1C(C(=O)NC2CC(C)(C)C2)CC1C)=O c1(OC)cccc(OC)c1C(=O)NC(C)(C)CC1CCCCC1 C12(CNC(C3(n4cc(-c5c(F)cc(Cl)cc5F)nn4)CC3)=O)CCCC1CC(=O)N2 c1(C(N2CC(NC(Cc3c(C)noc3)=O)C(F)CC2)=O)cc(C#N)ccc1Br C1(C(=O)NC2(C)CC2)CC(F)CN(C(c2cccc(C(C)(C)C)c2)=O)C1 c1(C(C)NC(=O)CC(C)(C)CNC(c2cn(C)nn2)=O)coc2ccccc12 c1(C(N2CCC(CN(C(Cc3cc(C)no3)=O)C)C2)=O)nccc2ccsc12 c1(C2C(C(=O)NC3(N4CCCC4)CC3)CC2)nc(S)n[nH]1 c1(C(N2CC(NC(=O)CC(F)F)CC(C)C2)=O)cc([N+](=O)[O-])cc2ccccc12 c1(CC)nc(C)ncc1C(N1CC2(C(=O)NCC3CCC(C)O3)CC1CO2)=O C(=O)(C1=CCCN(CCCC(c2ccc(OC(F)F)cc2)=O)C1)OC N1(C(c2c(C)c(C3CC3)on2)=O)CCC2(CC2NC(c2cnsc2)=O)C1 N1(C(CCC2CCN(C(C(C)c3cc[nH]n3)=O)C2)=O)CCCCN(C)CC1 C(=O)(C(F)C(C)C)N(CC(C)NC(Cc1nc(C(=O)OC(C)(C)C)sc1)=O)CC C1(C2(C(=O)OC)COC2)CCCN1C(c1ccnn1C1CCCCO1)=O CN(CC(=O)OCC1CC1)N1CCn2nc(COc3ccccc3)cc2C1 N1(C(c2c(C)ccc(F)c2)=O)CCC(F)(F)C(NCc2cc(F)c(F)cc2F)C1 C(=O)(C(C(CC)NC(=O)C(C)(C)c1ccnn1C)C(C)C)OCC N1(C(C(n2cc(COCC3CCCC3)nn2)C)=O)CCOC(CC2CCCC2)C1 C1(NC(c2cc(C)cc(Cl)n2)=O)CCC2CN(C(=O)CCC(N)=O)CC2C1 N1(CC)C(=O)CCC1CC(=O)NCCN(C1CCCCCC1)C(C1CC(C)C1)=O c1(C(=O)NCC2(CNC(c3c(C)nc(C)[nH]3)=O)CCC2)ccc2c(c1)CC(C)O2 c1(C(=O)NCC2(C)N(C(CNC(CC)=O)=O)CC(F)(F)C2)cc(S(C)(=O)=O)oc1C CN1CCC(C(=O)N(C2COCC2(C)C)C2CC2)CC1.C12(CCC1)CC(=O)NC2 c1(C(N2CC(NC(COCC#C)=O)C3C2C3)=O)ccc(-c2cccs2)cc1F CN1CCN(C(C2CCCSC2)C(=O)NC2CCOCC2)CC(C)(F)C1 C1(CCC#C)(NC(=O)OCC)CCCCC1.C1C(OC)CN1 N1(C(C2CNC2)C)CCC2C(C1)NC(=O)CCN2C N(C(=NCC(C)C1CCCCC1)NC(c1cccnc1)C)C(C=C)C C(=O)(N=c1nc[nH]n1C)C1N(Cc2cc(OC)ncn2)CC(O)C1 C1(CNC(Cc2c(C)occ2)=O)CC(NC(C23CC(F)(C2)C3)=O)CCO1 Cc1ccc2cccc(C(=O)NCCC3CCCCN3C(=O)C=CS(C)=O)c2n1 CC1CN(C(=O)COc2ccc(O)cc2)C(C)CN1C(=O)CCC(F)F c1(N2CC(C(C)NC(c3n[nH]c4ccccc34)=O)C2)cc2c(cn1)C(=O)CCC2 C1(CC)(CNC(c2nnn(C)c2C)=O)CCN(C(C2CC(N3CCCC3)C2)=O)C1 c1(C(C)(C)C)conc1C(=O)NC1CCC1NC(c1cncn1C1CC1)=O C12(CNC(CC(CC)O)=O)CCC(CC1)N2C(c1cc(Cl)ncc1N)=O S(=O)(=O)(c1ccc(C#N)c(NCc2nccn2CCO)c1)N(C)Cc1nccs1 C1(NC(C(C)NS(CCCC)(=O)=O)=O)CCCN(C(=O)CCCF)C1C N1(c2nnc(C)s2)CCC(C2CCCN(C(C3CCC4(C3)CC4(F)F)=O)C2)CC1 Cc1cc(C)c(NC(=O)C(N2CCC(C)CC2)=O)c(C)c1.OC(F)F C#CC1CN(C(C2C(CC)CCN2C(=O)CCc2cn(C)cn2)=O)CCO1 N1(C(c2cncc(SCC)n2)=O)CCN(C(=O)Cn2cccnc2=O)C(CO)C1 C1(NC(CCCSC(C)(C)C)=O)CC2(C1)CC(NC(c1cn(C3CC3)nn1)=O)C2 C1(CNC(C2C(COC)C2)=O)(CO)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1.C(C)(=O)O C1(CCn2cc(CN(CCOC)C(C3CC3C#N)=O)nn2)COCC(C)(C)O1 C1(C)(C(=O)NCC2(SC)CCC2)CCOCC1.c12ccc(s1)CC(=O)NC2 N1(C(C23CCC(NC(c4cc(C)ns4)=O)(CC2)C3)=O)CC(=O)NC(C)(C)C1 N1(C(C2(COCC)CC2)=O)C2CCC1CC(CNC(=O)C(C)C(C)O)C2 N1(C(C(CCC)OCC)=O)CCC(F)(C(=O)NCCN2CCC(OC)C2)CC1 c1(CC(=O)NCC(CNC(CCN(C)CC)=O)CO)cc(C)ccc1C C(=O)(CN=c1ccc(C#N)c[nH]1)NC1(CNC(CC(C)N(C)C)=O)CCC1 c1(CC)ccc(C(=O)NC2CC23CC(NC(c2cc(C(C)C)nn2C)=O)C3)cc1 C1(CNC(C2(C)C=CCC2)=O)CCCCN1C(c1sccc1-c1ccccc1)=O Cc1c(C)c(OC(c2cnc3c(c2)nnn3C)=O)c(C)c(C)c1C N1(C(C2C(C)(CC)C2)=O)CCCC(F)(C(=O)NC2(c3noc(C)n3)CC2)C1 C12(C(N3CC(CCC)C(CO)C3)=O)CC(C)(CN1C(c1ccoc1Cl)=O)C2 C(=O)(CCC(C)c1ccccc1)N1CC(=C(CNC(CC2CCC(C)C2)=O)F)C1 N1(C(C2C(C(=O)OCC)C2)=O)CC2CC(NC(c3ccn(C)n3)=O)C1C2 c1(C(N(C2CCCN(CC3(C#N)CCNC3)C2)CC)=O)ccc(Cl)cc1OC C1(CC(=O)NCC2C(CC(=O)N(CC(=O)NC)C)C2)OCCO1 CC(C)(C)CC(O)CC(=O)NC(CNC(=O)CCc1cccc(F)c1)CO C(CC(C)N=c1nc(C#N)[nH]cc1Cl)NC(C1CCCN(CC)C1)=O c1(C(=O)NCC(CC)NC(c2cn(CC(N)=O)nn2)=O)cc(F)ccc1Cl C1(NC(c2cncc(OC)c2C)=O)CN(C(=O)CC(F)(F)F)CC(C)(C)C1 C=CCCCCCCC(=O)NC1COCC1CNC(C1CCC2CC1C2(C)C)=O CCCC(CC(=O)N1CCC(N(C)C)C1)NC(C1CC(=O)N(OC)C1)=O N1(C(C2C(C)N(C)CC2)=O)CCCCC(CN=c2[nH]nc(C(N)=O)s2)C1 c1(OC)cnc[nH]c1=NCCc1cc(Br)no1 C1(F)(CNC(=O)C=Cc2ccco2)CCCN(C(C2CC23CC3)=O)C1 c1(C(=O)NCC2C3CN(C(CSSC)=O)CC32)nc(C(C)C)ncc1Br n1(CC)ncc(CNC(CC2N(C(=O)NC3CC3C3CCCO3)CCCC2)=O)c1C C1(C(=O)NC(CCOC)CO)CN(C(C2CC(=C3CCC3)C2)=O)CC12CC2 N1(C(c2c(C)nc(CC)o2)=O)CC2CCN(C(c3c(CC)noc3C)=O)CC2C1 Cc1cc(C(=O)NCC2(CNC(c3cncn(C)c3=O)=O)CCC2)ncc1Cl C1(COC)CC(CNC(=O)C(C)Cc2cccc(Cl)c2)N(C(=O)CCF)C1 C1(C2CC2)(NC(C2C(OC)C2)=O)CCN(C(c2cnc3n2CCS3)=O)C1 c1(C(C(=O)NCCC#N)N(C)CC2CCCS2)cc(Br)ccc1Cl c1(CCCC)oc2ccccc2c1CNC(C)CCNC(C1CSCCS1)=O C1(C(CNC(C2(C)CC2)=O)(C)O)CCCN(C(C2(c3ccccc3F)CC2)=O)C1 C1(NC(CC(C)c2ccco2)=O)(CNC(=O)C(O)Cn2cncn2)CCOCC1 c1(C(=O)NC2CN(C(C(CC)n3ccnc3)=O)CC2C)cnc(OC)c(CC)c1 c1(C(N(CC(C)NC(C2(F)CC=CCC2)=O)CC)=O)coc2c(F)cccc12 C(CC(C)CC)(C(=O)NOCc1ccccc1)NC(c1cc(CC)on1)=O C1(C(=O)NCc2nc(CC)on2)CN(C(c2cc(OC)n[nH]2)=O)C(C)(C)C1 N1C2CCC1(Cn1cc(C3(O)CCCCC3)nn1)CC2.O=C1CCCC(C=O)O1 C(CCc1cccs1)(C(C)NC(=O)CSC(F)F)NC(C1CC(C)C1)=O N1(C(c2c(COC)cco2)=O)CCOC(C(=O)NC2CCCC2OC)C1 Cc1cc(=NCC(=O)OC(C)(C)C)[nH]c(NCCS(=O)C(C)(C)C)n1 CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc[n+]([O-])cc2)=O)C(F)(F)C1 c1(NC(CC)CNC(=O)C(C)Cc2ccccc2)ncnc2n[nH]c(C)c12 N1(C(c2ccnc(Br)c2)=O)CC2(CCCCN(C(C3COC3)=O)C2)C1 Cc1cc(C=CC(=O)NCC2CC(C(=O)O)CCO2)ccc1C(F)(F)F c1(C(=O)NCC2(NC(C(C)(CO)OC)=O)CCOC2)cc(C)cc2ccncc12 C#CCCCC(C)C(=O)N1CCC(NC(=O)Cc2c(C)cccc2Cl)C1 c1(SCC)ccc(C(=O)NCC(C2CCN(C(c3c[nH]nc3F)=O)CC2)F)cc1 Cc1nc(O)[nH]c1C(=O)NCC1CCCCN1C(C1CCCCC1)=O C(=O)(CS(=O)(=O)C(C)C)NCC1CC(NC(Cn2cc(C(=O)NC)nn2)=O)C1 C=CCC(CNC(c1cc(C)cc(C)n1)=O)C(=O)NCC(Cl)C(C)(F)F c1(C(=O)NC2CCN(C(=O)C(F)=C3CCC3)CC2)cncc(Br)c1Cl c1(NC(C(COC)(C)C)c2nnnn2C)cc(F)ccc1CC.C(C)(C)(C)NC(=O)OCC N1(C(CC=CC(C)(C)C)=O)CCCC2(CCCN2C(=O)CCCF)C1 C(C(C)CC(=O)NC(Cn1cncn1)C(N1CCCOCC1)=O)OC C1(C(N2CC(c3cn(CC(C)C)nn3)N(C)CC2)=O)CCc2nccn2C1 c1(C(N(C(C2CC2C2CC2)C(=O)NC(C)C)C)C)cccc(Cl)c1 CCCCC(F)C(=O)N1CC(CNC(C2(C(F)F)CCCO2)=O)C2(CC2)C1 c1(C(N2C(CN(C(C3OCCN(CC)C3)=O)C)CCC2)=O)cnc2scc(C)n12 CC(C)(C)CCCCC(=O)N1C2CCC1CC(O)(CNC(c1cc(F)n[nH]1)=O)C2 O=C(N=c1ncn(C2CC2)[nH]1)NCCOCCCO.C(CS)NC(=O)C1CC1 CN=c1cc(C(=O)NC23CCN(C(c4oc(C(C)C)nc4C)=O)CC2C3)cc[nH]1 c1(N2CCN(C(c3cc(CC)[nH]n3)=O)CC2CC(C)(C)C)nc2ccccc2o1 c1(N2CCCN(C(C(C)C)=O)CC2)ncnc2c1ncn2C1(CO)CCC1 C(=O)(C(C(C)C)NC(=O)C=CCC(C)(C)Cn1cc(-c2ccccc2Cl)nn1)OC c1(C(=O)NCC(=O)OCCCC)ccc(CNC(=O)C(C)n2cnnn2)cn1 N1(C(c2c(C)cc(Cl)cc2)=O)CC(N=c2[nH]c3cccc(C)c3o2)C1 C1(c2n(C(CC)C)nnn2)(NCc2noc(C3CCCC3)n2)CC2CCC(C1)O2 CCCC(CNC(=O)CSc1ccccc1Cl)CCC c1(C(=O)Nc2ccc(NC(C3CC=CCC3)=O)nc2)cc(Cl)ccc1Cl c1(CNC(N)=O)ccc(C(N2CC(NC(C3CCCCC3)=O)C3CC23)=O)cc1 C(C(C)C)(C(O)C(=O)N1C(CC(N2CCC(C)C(C)C2)=O)C2CCCC12)OC C1(C(=O)NCC2CCN(c3ncc(C(=O)OC)s3)C2)CC(C)OC1C Cc1noc(CCCC(=O)NCC2CCCC2NC(=O)C=Cc2cc[nH]c2)n1 Cc1ccc(C#N)cc1CCSc1ccc(C(F)(F)F)nc1C CC1=C(C(=O)N2CC3C(CN(C(=O)CC4SC(=N)NC4=O)C)C3C2)CCO1 C1(C(=O)OC)C=CC(C(=O)NC2CC(N(C(=O)C=CC3CCCC3)C)C2)C1 N1(Cc2nc(C)c(C)s2)CCOCC1(C)C.N12CCCC1NC2=O C(CC(C(C)(C)C)NC(=O)CC1(C)CCOCC1)N(C)C(c1cc(O)cs1)=O C(CC(C)C(=O)N(C)CC1CN(C(c2cc(Br)cn2C)=O)CCO1)=CC c1(N(C)C)ccc(C(N2CC(COC)(NC(=O)CC(C)CN(C)C)C2)=O)cc1F C1(NC(c2cnc[nH]2)=O)CC2CC1CN2C(=O)CCc1ccccc1Cl C(C(=O)N1OC2CCC1C2)C(C1(CC(=O)NOC2CCC(O)C2O)CC1)C N1(C(Cc2ccc(C)cc2)=O)CCC2(CCC(C(=O)NCC(C)CO)CC2)CC1 Cc1cc(C(=O)NCC(CC2CC2)C(=O)NCc2cccnn2)nc(O)n1 CCCC(CCCNC(=O)CCc1ncc[nH]1)NC(C1(CN(C)C)CC1)=O N1(C(C(c2ccc(C)cc2)=O)=O)CCN(C(=O)CC2OCCC2C)C(C)C1 Cc1cc(NC(C2CCCCC2NC(C2(C)CC(C(F)(F)F)C2)=O)=O)cc(O)c1 C1(C(N2CC3CC(NC(CC(C(C)C)C)=O)C3C2)=O)CC2(C1)CC(F)(F)C2 c1(C(=O)NC2CC(CC(=O)NCCCC(C)OC)C2)ccnc(CN(C)C)c1 C12(CNC(=O)CC3CCOC3)CC1CN(C(c1cc(Cl)c[nH]1)=O)C2 C1(C(=O)NCCCCCNC(C2CCC(CN(C)C)O2)=O)CCc2nccn2C1 c1(OC)noc(C)c1C(N1CCCC(CCNC(=O)CC2CCCN2C)C1)=O c1(C(N)=O)csc(C(N2CC(NC(C3COC(=O)C3)=O)C2)=O)c1 CCCC(C(=O)NCc1ccc(CNC(=O)CC2C=CCC2)cc1)NC(N)=O N1(C(CNC(=O)OC)=O)CC2CCN(C(c3ccccc3)=O)C2C1.C1(N)CC(C#N)C1 c1(C(N2CCC(C(C)NC(CC(CCC)C)=O)C2)=O)ccc2nc(C)cn2c1 C12CC3CN(CC3C1)C(=O)c1ccc(o1)NC2=O.C1(C(N)=O)CCCC(N(C)C)C1 c1(C(=O)NCCC2(NC(CN(CC)CC)=O)CCC2)cc(CO)oc1C C1(NC(C2C=CCN(C(C(C(C)(C)C)OC)=O)C2)=O)CN2CCC1(C)CC2 N1(C(Cc2cn(C)nc2)=O)CC2CC(NC(=O)C3=NNC(C(F)(F)F)C3)C2C1 N1(CCOC)CC2(CN)CC1(c1nc(-c3nc(C(=O)OCC)c(Br)s3)no1)C2 N1(C(CCn2c(C)ccc2C)=O)CCC(CCNC(=O)CC(C)C2CC2)CC1C C12(F)CCN(CC1)C2=O.c1(C(N2C(C(=O)OC)C=CC2)=O)cnc(C2CC2)cn1 C1(CNC(C2CC(C)OC2)=O)C2CC1N(C(=O)Cc1ccccc1Br)C2 N1(C(c2c(C)scc2)=O)CCC2(CC1)CCN2C(c1cocn1)=O c1(OC)ccc(C(=O)NC2CC2CC(C)(C)C)cc1NCc1ccc(Cl)s1 N1(C(Cn2ncc(CC)c2)=O)CCN(C)C(CNC(C23CC(F)C2C3)=O)C1 N(C(=NCC1CCC1)NC1CCOc2ccc(F)cc21)CC1(SC)CCOCC1 c1(NC(c2nnnn2C2CC(F)(F)C2)(C2CC(F)(F)C2)C)ccc2nsnc2c1 N1(C(C2(CC)CC(C)(C)C2)=O)CCCC(CCNC(c2nncs2)=O)CC1 C1(NC(c2nc(COC)oc2)=O)CC2CC(NC(=O)CC(C)SC)CC2C1 N1(CC)CCCC1C(N1CC(NC(c2[nH]nnc2-c2ccnn2C)=O)C1)=O Cc1cnc(CNC(=O)C(C2CC=CCC2)NC(=O)Cn2ccnc2C)c(F)c1 n1(CC(=O)NCC2C(C(=O)NC3CC(C(C)(C)O)C3)CCO2)cccnc1=O C1(COC)(NC(C2CCOC2C)=O)CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1 N1(C(COCCC#C)=O)C2CCC1C(CNC(=O)Cc1c(F)cncc1Cl)C2 N1(C(CCNC(C)=O)=O)CC2CN(CCc3ccc(Cl)cc3)CC2C1 N1(C(C(C)C(C)(C)C)=O)CC2CCN(C(c3c[nH]cc(F)c3=O)=O)CC2C1 c1(C(=O)O)cc(Nc2ncnc3c2SCC3)cc(F)c1F c1(CC(=O)NC(CNC(C2C(CCC)C2)=O)(C)CO)sc(C)cc1Br n1(CC(C)Sc2cccc(F)c2)nc(-c2ccoc2)nc1C1CCc2cccnc21 C(=O)(C1CC(=O)Nc2ncccc21)N1C(CNC(C2N(C(C)C)CCC2)=O)CC1 N1(c2c(C(=O)NC)c3c([nH]2)cccc3)C(=O)c2ccccc2C1=O c1(CN(CP(=O)(OCC)OCC)CCOCC#C)cn2cc(Cl)cc(Cl)c2n1 C1(CNC(c2ccn(C)n2)=O)CCCCCN1C(C1CCCN1CCC#N)=O C1(C(=O)NC(C(CC)C)CO)C2CC(O)C(C2)N1C(c1ccsc1C#N)=O CC1CN2CCN1CC2C(N1CCC(C(C)Nc2ncnc3c2CCC3)C1)=O C(=O)(C(C)(C)CN(C)C(C1CC2(CSC2)C1)=O)N(CC(CC)CC)CC c1(C(=O)NCC(CC=C)NC(c2n[nH]cc2Cl)=O)ccc(C(C)(F)F)nc1O CC1=C(C(=O)NC2CCCN(C(=O)C(N3CCC(C)C3)=O)CC2)C(=O)OC1(C)C c1(C(=O)NC2CCC(NC(c3c(C)nn(C)c3)=O)C2)c[nH]cc(F)c1=O C(CCNC(=O)C(C1(O)CN(C(=O)COc2ccc(C)cc2)C1)F)(C(C)C)OC CN1N=CC(CC(N2CCC(C(F)F)(CNC(c3cc(=O)n(C)o3)=O)C2)=O)C1=O N1(C(C2(C)N(C(CCCC)=O)CC=C2)=O)CCC(C)OC(C)C1 N1(C(COCCCCC)=O)CCCC12CCCN(C(C1CC(F)C(=O)N1)=O)C2 Cn1ccc2cccc(C(N3C4CCC3CC(NC(C3CC3(F)F)=O)C4)=O)c12 C(C(C)(C)CCNC(c1cn(C)cn1)=O)NC(C(C)OCCCCCC)=O N1(C(CC(COOCC2CC2)NC(C(CC)CCOC)=O)=O)CCc2nncn2CC1.OC c1(SCCCC)ccc(C(=O)NCC2(F)CC(NC(C3(F)CC3C)=O)C2)cc1 N1(C(C2OCCN(CC)C2)=O)CCCOC(CCNC(C2CCCC2)=O)C1 CCC(C)(CC)CN=c1nc2scnc2c(NCC2(C)CCCCO2)[nH]1 N1(C(Cc2ccn(CCOC)n2)=O)CCC(NC(=O)CNS(N)(=O)=O)CC(O)C1 C1(C(N(CCNC(C2C=CCCC2)=O)CC)=O)CC2CCC(C1)O2 C(=O)(C1=CC2(CCOC2)C1)NCC(CC)(CC)C(=O)NC1CN(C)CCC1O N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)CC(C)C2CCCCC2)CC(CO)C1 C1(NC(C2N(CC)CC2)=O)CCCC2CN(C(c3cn(CC)nc3C)=O)CC12 c1(NC(COC(CC)C)=O)cc(COC)ccc1[N+](=O)[O-].C12(CC1)C(=O)NC2 C1(NC(C2N(C(C)=O)CCC2)=O)CN(C(C2(CC(C)C)COC2)=O)CC(C)(C)C1 c1(NC(c2cn(CCNC(=O)Cc3ccns3)nn2)=O)cccc(C2CC2)c1 CCCCC(C)(F)C(=O)N1CCCC(CN(C)C(c2cc(C)nc(O)c2)=O)C1 Cc1cc(C(N2CCCC2c2cn(CC3CCC(=O)O3)nn2)=O)cc(C)c1C O=C(NNc1ncc(I)cn1)C1CCCN(CCC2CCCO2)CC1 c1(N(C)CC2CCN(C(Cc3c(C)ccc(Br)c3)=O)C2)cc2nncn2c(C)n1 c1(OC)ccccc1C1CNCCN1C(N1CCC(CF)C1)=O C1(NC(C2(C(C)C)COC2)=O)CCC2CC1CN2C(=O)CC1CCCNC(=O)C1 N1(C(c2c(C)n(C3CC3)nc2)=O)CCC(CNC(=O)C(F)CC2CC2)C(F)(F)C1 c1(C(C(=O)NCCOC)N(C)CC2CC2)nncn1C CC1CCCC(C)N1C(=O)C(=O)NC1CC(N(C)C(c2cccnc2)=O)C1 C1(C(=O)NCC2CCC2(F)F)(NC(Cc2c(C)occ2)=O)CCN(C)C1 Cc1ncc(C(=O)NCC2(C(C)(C)O)CN(C(C3(C)CC3F)=O)C2)s1 c1(C(N2CC(C)C(NC(=O)CCCCF)C2)=O)cccc2nc(O)oc12 N1(C(c2c(N)ccc(C)c2)=O)C(C)CC2CN(C(C3(C)CC3(Cl)Cl)=O)CC12 C1(CC(=O)NCCN(C(=O)C=CC2CCOC2)CCOC)CCCC2CC12 C(=O)(CCCCCNC(C1C2COCC12)=O)N1CC(=CCC)C1 C1(NC(C(=O)NC(C)C)=O)CCN(C(c2cc3nnn(C)c3s2)=O)CC(O)C1 CC#CCCCC(=O)N1CC(C(N)=O)(CNC(=O)C(C)(F)F)C1 C1(NC(=O)C(F)n2ccnc2)CCN(C(C2CC2(Cl)Cl)=O)CC1 C1(C)(COC(C(c2cn(C)nc2)O)=O)CCCC(F)(F)C1 c1(C(=O)NC(CNC(C(C)=C(C)C)=O)CO)cc(F)ccc1Br c1(C(=O)NC2C(NC(c3c(CC)nns3)=O)CCC2)ccc(Cl)c(O)c1N CCC(C)(CNC(c1nnn(C)c1N)=O)C(=O)NCC(O)CCC#N C1(NC(CN2CC(C)C2)=O)(CNC(C2(C(F)(F)F)CC(O)C2)=O)CCCCC1C CC1(C(=O)NC2CC(C)(NC(c3ccc(CO)cc3)=O)C2)CC(C2CC2)=NO1 C1(CNC(=O)C(C2(O)CN(C(=O)C(c3cccnc3)O)C2)F)C2(CC2)C12CC2 N1(C(C(=Cc2cnc[nH]2)C)=O)CCCC(C)C1CNC(c1nccnc1C)=O CC1C(NC(=O)N(C)C)CCCN1CCCN1CCCC1=O C1(c2cc(C)cc(C)c2)CC2(CCOCC2)C1.c12ccccc1COC2=O C(=O)(CC(C)C(=O)c1ccccc1)N(C(CNC(c1c(OC)ccs1)=O)C)C C1(CC)CC(C(=O)NCc2cc(C3CCN(C(=O)C4=CCC4)CC3)no2)CCO1 CCCCC(C)C(=O)N1CCC1CNC(=O)C(C)Cc1c(C)noc1C Cc1ccc(C(N2CCN(C(=O)CC3(C)CCOC3)CC2CCO)=O)c(=O)n1C S(=O)(=O)(c1nc(N2CCC(C(F)F)CC2)ccc1Br)NCC(C)(C)c1cccs1 c1(CNC(C(=O)NCC2(CCl)CC(C(CC)C)C2)=O)nsc(C(=O)OC)n1.CC N1(C(c2cnn(CC(F)F)c2)C(=O)NCCOC)CCC2(CCOCC2)C1 C1(CCNC(C(C)NS(C)(=O)=O)=O)CN(c2ncc3c(n2)COC3)CCS1(=O)=O c1(C(N2CCCC(CNS(=O)(=O)Cc3ccccc3Cl)C2)=O)nccc(Br)c1O C(=O)(CC(O)CC(C)(C)C)N1CCC(N(c2ccccc2Br)C(C)=O)C1 N1(C(C2(C(N)=O)CCC2)=O)CCCC(n2cc(-c3ccc(C(=O)O)nc3)nn2)C1 C1(CNC(C2(CC)CC2)=O)CC(C)(C)CCC1NC(=O)C=Cc1ccc(C)cn1 CN1CCN(C2CC(CNC(N3CCC(CCO)(CN(C)C)C3)=O)C2)CC1 CC(C)C(N=[N+]=[N-])C(=O)NC1CC1CNC(C1CCOC1c1ccnn1C)=O C1(NC(=O)C(Cl)=CCl)CCCCC12CCN(C(c1coc(Cl)c1)=O)C2 C1(NC(CCCc2cc(C)no2)=O)CCN(C(=O)COCC2CC2)CC1C N1(C(=O)Cc2cccs2)CCC(C2CCCN(C(c3ncoc3C(F)F)=O)C2)C1 CCC(C)(CCNC(C1CCSC1)=O)NC(=O)C(O)CSC N1(C(CCOCCC)=O)CCC2(CNC(c3cc4c([nH]3)CCC4)=O)CCCCC12 CC1CC(C(N2CC(C3(NC(=O)C#CC4CC4)CC3)C2)=O)CCS1(=O)=O C1(C(=O)NC2(C)CC(NC(=O)C3=CCCC3)C2)CCCC(F)(F)C1 N1(C(c2cc(OCC)cc(CC)c2)=O)CCCC(C2CC2)CC1 C1(C(=O)NCC2CCN(C(CCOC(C)=O)=O)C2(C)C)CCC2(CC1)CC2(F)F C1(CC(=O)NCCN(C(C(F)=C(C)C)=O)C(C)C)CC(=O)NC1=O N1(C(C(CCC)CC)=O)CCCC(C)(C)C1CNC(C1CCN(OC)CC1)=O c1(C(=O)NCC2CC3N(C(C4C(C#N)C4)=O)C(CC3)C2)ccc2oc(O)nc2c1 N1(CCC)C(=O)CCC1C(=O)N(C(C)CNC(C1CC(C#N)C1)=O)C C1(CN(C)C(c2cocc2Br)=O)CCN(C(c2scnc2C2CC2)=O)C1 S(=O)(=O)(CC(=O)NCCCN1CCN(C(C2CCCC(OC)C2)=O)CC1)NC c1(N(C)C(=O)OC(C)(C)C)ccc(NC(=O)NCC2(F)CC2)cn1 c1(C(N(CCC)CCNC(=O)C(C)CC)=O)noc(C)c1I c1(CNCCC(CCO)N(C)C)cccc(C(F)(F)C(F)(F)F)c1 CCC(C(=O)NCC1C(C)CCN1C(=O)C(c1n[nH]c(C)n1)NC(C)=O)C(C)O C(=O)(C(C)(C)COCC)N(CCC)CCNC(C1CC=CCC1)=O c1(C(N2CCCN(C(C3CCC34CCCO4)=O)CCC2)=O)cc2cccnn2n1 c1(C(N(CCS(CC(C)C)(=O)=O)C2CNC2)=O)cc(=O)n2nccc2[nH]1 N1(C(C2=CCC(NC(C3(C)CCCO3)=O)C2)=O)CCN2CCC1CC2 N1(C(c2c(C)noc2)=O)CCCC2C1CCN2Cc1cccc(C(N)=O)c1 C1(C(N2CCC(N3CCN(C(C4C(C)CCC4)=O)CC3)C2)=O)CN2CCN1CC2 C1(NC(C(C(CC)C)C)=O)CC2(CCC(NC(C3CC(C)CCO3)=O)CC2)C1 N1(C(COC)=O)CCCC(OCc2cn(CCCF)nn2)C1 n1(CC(N2CC(C)N(C(c3ncccn3)=O)CC2)=O)sc2ccccc2c1=O N(C(=NCCOC(C1CCCCC1)OC)N1CN(C)C(=O)C1C)C(C=C)C C1(NC(COCC)=O)CC(F)CN(C(=O)C(C2CC2)Sc2ccccc2OC)C1 N1(C(C(CCOC)C)=O)CCC(NC(c2ccn(C(C)(C)C)n2)=O)C(F)(F)CC1 Cc1ccc(C=CC(=O)N(C)CC2CN(C(=O)CNC(C3CCC3)=O)CCO2)s1 C1(N(C)Cc2ccc(NC(C)=O)s2)CCN(C(=O)CO)CC1.C1(CC2CC2)CCCC1 N1(C(C(C(C=C)C)C)=O)CCC2(CC1)CN(C(C1CN3CCN1CC3)=O)CCO2 N1(C(CC2(OCC)CCC2)=O)CCOC(CNC(C2CCC(CC#N)CC2)=O)C1 C1(CNC(C=CC)=O)CC2(CCN(C(C3CN(C)CC3C(F)(F)F)=O)CC2)C1.NC c1(NC)ccc(C(N2CC3(CCC3NC(=O)C(C)SC(F)(F)F)C2)=O)c(Cl)c1 N1(C(c2c(CC)oc(C)c2)=O)CCCC(O)(CNC(C2CCCC(C)CC2)=O)C1 c1(N2C(CC#N)CN(C(C3CSCC(=O)N3)=O)CC2)c(F)cc([N+](=O)[O-])cc1F N1(C(C=CC(c2ccc(Cl)s2)=O)=O)CC(NC(C2CC(=O)N2)=O)C(C2CC2)C1 c1(CCC(=O)NCC(CN(C(C(C(C)C)C)=O)C)C)ccc2c(c1)CCCO2 C(CC(C)C(=O)N1CC(CCNC(c2cnsn2)=O)(OC)C1)=CCC C1(N(CC(C)C)C(c2onc(CCC)n2)=O)CCN(C(N2CCC(C)C2)=O)CC1 C(=O)(C1=CC2(CCOC2)C1)N1C(CNC(CCC(=C)Br)=O)COC(C)(C)C1 S(=O)(=O)(c1nc(N2CCC(C)(F)CC2)ccc1Br)N(CC(C)OC(C)(C)C)C O=C(N=c1cc(-c2cccc(F)c2)[nH][nH]1)c1cnn(CCCOCCO)c1 C(=O)(C1=CC2(CCOC2)C1)N1C2CC(C(N3C(C(=O)NC)CC3)=O)CC1CC2 C1(NC(C2CCCCC2)=O)COCCN(C(=O)CCOC2CCOCC2)C1 C1(C(=O)NC(C)CN(c2nccc(COC)n2)C)(COC)CCOCC1 C(=O)(C(=O)C(C)(C)C)N.C12CCC(C1)NC(=O)CC1(CC1)C(=O)NCC2.CSC c1(C(C)C)nc(C(=O)NC(C)C(C)NC(c2nc(C3CC3)cs2)=O)co1 c1(C(N2CC(N(C(C(CC)CC)=O)C)C2)=O)c(-n2cccn2)cccc1F CCCCS(=O)(=O)N1CCCC(C(N2CC(NC(c3cnn(C)c3N)=O)C2)=O)C1 C1(C(N(CC(C)NC(c2ccsc2OC)=O)CC)=O)CN2CCCN1CC2 C1(c2n(C)nc(-c3cc(F)cc(F)c3)n2)CC12CCCOC2 CC(C)(C)C(CNC(=O)CC1CC2(CCC2)C1)NC(C1CCC=CCC1)=O C1(C(=O)NC(CC=C)CNC(c2ccc(Cl)c(OC)c2)=O)CC2C=CC1CCC2 C12CC=CCN1C2=O.C1(C(N2C(C(=O)OC)CC2C)=O)C2CC3C(C2)C13 c1(C(=O)NC(C)CNC(=O)CN2CCC(C)(O)C2)cccc(F)c1Br C(=O)(C1=C(C2CCC2)N(C2CC2)C(=O)NC1c1noc2c1CC(F)(F)CC2)OCC c1(C(=O)NC(C2CCN(C(=O)CSc3nncn3C)C2)C)ccn2ccnc2n1 c1(C(=O)NCCN(C(Cc2c(C)ncs2)=O)CC(C)O)c[nH]c(C#N)c1 c1(C(N(C(C)CCNC(C2CC(C)(F)C2)=O)C)=O)ccc(-n2ccnc2)cc1 n1(CCC)nnnc1C(c1sccc1C)NCC=CCl c1(C(=O)NCCC(CC)O)cc(Cl)cc(COC)n1 CCCCCCC(=O)NCC(C1CCN(C(=O)C(C)(C)C2CCCO2)CC1)C N#Cc1ccnc(C(=O)NC(C2CC(F)(F)C2)CO)c1F c1(C(N(CC(CNC(C(C)OCCCC)=O)C)C)=O)c(C)nn(C)c1OC C1(CCC)(NC(CCCC=C)=O)CCCN(C(=O)C(CC)N2CCCC2=O)C1 C(=O)(CCCC(F)(F)CO)N1CC2C(CNC(c3cnn(C(C)C)n3)=O)C2C1 CC1(C)CN(S(=O)(=O)CCN(C(=O)C(Cl)Cl)C2CC2)C1=O n1(C(C)C)cc(C(N2CC(O)(CN(C(=O)C(C)(C)c3cccnc3)C)C2)=O)cn1 Cc1ccsc1C=CC(=O)OC.c1(COC2C3(CCC3)NC2)ccccc1 C#CCCCC(C)C(=O)N1CCOC(C(N2CCN(C(=O)CC)CC2)=O)C1 C1(CNC(c2cc(C)oc2C)=O)(CO)CCN(CCn2cc(Cl)cn2)CC1 C1(CNC(C(=O)N(C)C)=O)CCC2(CCN(C(c3ccsc3S(C)(=O)=O)=O)CC2)O1 C(=O)(CCCCc1ccc(Cl)cc1)NCCC(C)N(C(C1N(CC)CC1)=O)C C1(C(=O)NCCNC(c2ncc[nH]2)=O)CCCCN1C(=O)C(O)CN1CCCC1 c1(C(=O)NC2CCC(NC(c3cccc(OCC#C)c3)=O)C2)cncc(C)c1C C(C(C(=O)N(CCNC(=O)CCC(C)CC)CCOCCO)C(C)(C)C)OCC=C N1(C(CCCCCC)=O)CCC2(CC2)CC1C(=O)NC1CCCOC12CCC2 N1(C(C2CCC2COCC)=O)CC2C(CO)C2C1.C12(CCC1)C(=O)NC2 c1(C(=O)NC2CCC2COC)ccc(CO)o1.C(=O)(COCCN)OC C(C)(C(=O)N1C2CCC1(CNC(C1C3CCCC13)=O)CC2)(C(C)C)NC(C)=O CC(CCCNC(C1CCCN1C(=O)C1CC1)=O)NC(c1cc(Cl)ns1)=O N1(C(c2c(C)cc[nH]2)=O)CC2CCCC2(NC(c2c(NC(C)=O)c[nH]c2C)=O)C1 C12(C(N(CCC)CCNC(C3C(C)(C)C3(C)C)=O)=O)CCCC1C2(F)F C=CCC(CC=C)NC(=O)CC1CCCC1NC(c1occc1C(C)C)=O N1(C(C2N(C)CC(OC)C2)=O)CCN(c2ccc(N(C)C)cc2)C(=O)C1 CCCN=C(NCC1CC2C=CC1CC2)N1CCN(C(c2ccccc2)C)CC1 N#CC(C(=O)CCc1ccsc1)C1CCCNC1=O.C1CCCO1 N1(C(C(C)NC(CC)=O)=O)CCCC1C1(C(=O)N(C(C)CC(C)C)C)CC1 C(=O)(C1=CC(O)CCC1)NCC=CCNC(c1ccc(C)c(Br)c1)=O c1(CS(N2C(C(N3CC4CCC3CO4)=O)CC(O)C2)(=O)=O)ccc2c(c1)OCO2 N1(C(c2c(C)n(C)cn2)=O)CCN(C(C2CC2C2CCC2)=O)CC1C(F)F c1(OC)cc(C(=O)NC2(CC(=O)Nc3cc(OC)ccc3Br)CCC2)ccc1O N1(C(=O)O)CCOC2(CCC2)CC1.c12ccc(F)c(c1)C(P(C)(C)=O)n1cc-2nn1 CCC(C)(C(=O)NC1CCCN(C(c2cc(C)c(CO)cn2)=O)CC1)C(N)=O c1(C(N(C2CCOCC2)CC#C)=O)cnc(CNC(=O)CC2COC(=O)C2)nc1 c1(OC)ccc(C(=O)NC2(CN(C)C(C3CN(CP(C)(C)=O)C3)=O)CC2)c(F)c1 C1(C(=O)NC(C=C)C)CCC(C)(NC(=O)C=CC(=O)OCC)C1 c1(C(Cc2ccccc2)N(C(CC)CO)C(C)=O)nnc2ccccn12 C12(C(=O)NCCC3(CNC(CC4N(CC)CCCC4)=O)CC3)CC=CC(C1)OC2 Cc1nn(C)cc1C1=NOC(C(=O)N(C2COC2)CCc2cccs2)C1 C1(N(C(C(CC)OC)=O)C)CCCCC1NC(=O)CCc1cc(OC)no1 C(C(C(=O)N1CCC(C(N2CCC(CC(C)(C)C)CC2)=O)O1)N(C)C)OC c1(OCC)cc(NC(=O)CCC=Cc2ccccc2)c(Br)cn1 N1(C(CN(C(C)C)C)=O)CCC2CC2(C(N2CCCCC(C)(C)C2)=O)CC1 C1(NC(C(C)OCCC=C)=O)CN(C(c2nc[nH]c2C(F)(F)F)=O)CC12CC2 N1(C(CC2N(C(c3n(CC)c(O)nc3)=O)CCC2)=O)CC2CCC(C1)O2 C1(N(CCCC)C(=O)CN(C)C)CCN(C(=O)C(CC)NC(=O)COC)CC1 C1(CNC(C(c2ccccc2)OC(C)C)=O)CC2CCC1N2c1nnn(C)n1 C1(C(=O)NC2CCCCC(I)CC2)C2CCCCCC12 c1(CC)cc(C)c(C(=O)NC2CCCC2C(=O)NC2(CSC)CC2)o1 C1(CC(=O)N(C(CNC(C(C)OC)=O)C)C)CCn2cncc2C1 CC1C(C)N(C(=O)C(C)(C)O)CCN1C(=O)C=Cc1cc(Cl)cc(Cl)c1 N1(C(C(CCC)C)=O)CCN(Cc2cccc3c2CNC3)CC12CC2 C12(NC(CC3CC(C)C3)=O)CCN(C(c3cnc(N)cn3)=O)CC1C2 c1(C(=O)NCCC2CCN(C(C(COC)(F)F)=O)C2)cc2c(C)nn(C)c2s1 CC1(C)CCC(NC(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)O1 C(C#Cc1ccccc1)NC(NC(CC)C)=NCCC1CC(C)(C)CO1 C1(NC(c2cnc[nH]2)=O)C2CC1CN(C(c1ncccc1CO)=O)C2 C1(CNC(c2c(N(C)C)nccc2)=O)CN(C(C2CC3CCC2O3)=O)CC12CC2 C1(C(=O)NCCCNC(=O)CCC2CCOC2)CCCN(CC(F)F)C1 C1(C(C)C)N(C(c2cnco2)=O)CC12CCN(C(c1ccnc(F)c1F)=O)CC2 CCC(CCCO)NC(C1C2CC1N(C(C1(OC)CCC(C)C1)=O)C2)=O C1(CC(=O)NC2CC(Cl)C2)Cc2ccccc2NC1=O CC(C)CCC(=O)NCC1(F)CC(CNC(c2conc2C(F)(F)F)=O)C1 c1(CC(=O)NC(CN(C(c2cnccn2)=O)CC)C)ccc(C)s1 N1(C(=O)C(O)c2ccco2)CCC2CCCC12C(=O)NC1CC2(CCCCO2)C1 c1(SC)cccc(F)c1C(=O)NC1CCN(C(c2nncn2C2CC2)=O)CC1C C1(C(=O)NCC2(C(N)=O)CN(C(CSC)=O)C2)C(C)OC(C)C1C C1C(C(C)C)C(=O)N1.C(C1=CCCN(C)C1)NC(C1(CC)CC1)=O N1(CC#C)CCN(C(=O)C(C)C(C)NC(c2occc2COC)=O)CC1=O C(=O)(CC(C)(C)C(F)F)N1CC(C(N2CC3CCC3(CO)C2)=O)CC(C)C1 C1(NC(CCS(=O)(=O)NC)=O)CC2CC(C1)N(C(c1cc(C)c(C)s1)=O)C2 C12(NC(c3c(C)oc(C)c3C)=O)CCCC1N(C(=O)CCOCC(F)F)CC2 C1(=O)C(CCC(=O)O)O1.C1(C)(C(=O)OC)C=CCCN1C(=O)OC(C)(C)C C(=O)(C(C)CNC(=O)CN(C(=O)C=Cc1cocn1)CCOC)OCC C1(C(=O)OCC)OCCNCC1N(C(=O)CCC1CCC1)Cc1occc1C N(C1c2ccccc2CC1NC(=O)CCCc1cc[nH]n1)C(C(CC)OC)=O c1(CC(=O)NC2CC(C)(C)N(C(=O)CC3CC3)C2)ccc2c(c1)COC2 CC1C(C(=O)N(C2CCCCCC2O)C)CCCN1C(c1cc2n(n1)CCO2)=O C(=O)(C1=NN2CCC(C)N=C2N1)NC1C(NC(c2cc(C)n(C3CC3)c2C)=O)C1 C(CCC(=O)NC1(C(=O)N(c2ccncc2)C)CC1)OCC c1(C(=O)NC2(C(C)C)CCNCC2)ccc2c(c1)ncn2C C(=O)(C(F)C(C)CNC(=O)CC1(O)CCOC1)N1C(C(=O)NC)CCCC1 C1(CNC(C(C(C)C)C)=O)(NC(=O)CNC(c2cscn2)=O)CCCCC1C C1(C(N2CC(C)N(C(c3n[nH]cc3Br)=O)CC2)=O)CCc2nn[nH]c2C1 C(=O)(C(=O)C(C)(C)C)NC(CNC(C(c1ccc(CCCC)cc1)C)=O)C(C)C Cc1ccc(C=CC(=O)NCCCC2CN(C(C3(C(C)C)CC3)=O)CCO2)nc1 c1(C(N2C(C)CC(NC(C3CCC(=O)N3)=O)CC2)=O)nccc2ccccc12 n1(CC(=O)N(C2CCN(c3nc(CC4CC4)ns3)C2)C)ccc2cc(F)ccc12 C(=O)(CCCN(C)C)NC1(C(N(C2(CC(C)C)CC2)CC)=O)CCC1 C1(OCC(=O)NCC(C)NC(=O)Cc2cc(C(F)(F)F)co2)CCCCCC1 C1(CC(=O)NCCCC2(NC(c3ccoc3C3CC3)=O)CC2)CCC(O)C1 C1(CCCC)(C(=O)NC(CC)CNC(=O)CC2CCCO2)CCCCC1 C1(C(N2C(C(=O)Nc3cn(CC)nc3C)CC3CC23)=O)(CC)CCOCC1 C1(c2n(C(C)C)nnn2)(NCC(=O)NC2CC(O)C2)CC(C)S(=O)(=O)C(C)C1 C1(C(C)C)CN(C(=O)C(C(C)O)NC(C2CC(=O)NC(=O)N2)=O)CC(=O)N1 Cc1ccc(C(=O)NC(C)CCCCNC(c2c(N)cnn2C)=O)c([N+](=O)[O-])c1 C1(c2n(-c3ccn(CC)n3)nc(-c3cccc(Cl)n3)n2)CCc2n[nH]c(C)c2C1 N1(C(c2ccnc(OC)c2F)=O)CC(NC(=O)CCC(C)N(C)C)C2CCCC12 CCC(C)(COC)C(=O)NCC(C)CN(C(=O)CCCN1CCCC1)C c1(C(=O)NC2C3CN(C(CNC(CNC(C)=O)=O)=O)C2C3)ccccc1S(C)=O CC(C)(F)C(C)(F)C(=O)NC(C)(C)CCCC(=O)NCCN=[N+]=[N-] C1(NC(C(C)NC(COC)=O)=O)CCC(C(=O)NC2CCC(C)CC2)CC1 C(=O)(CCCCCc1cccs1)N1CC2C(NC(C(C(C)C)OCC)=O)(C2)C1 c1(C(=O)NCC(CNC(c2cccc(C(C)C)n2)=O)F)cnc(O)c([N+](=O)[O-])c1 C12(C(=O)OC)CCCCCC1N(C(=O)NCCOc1ccc(Cl)nc1I)CC2 c1(CC(=O)NC2(CC(=O)N(CCCCC3CCCC3)C)CC2)ccccc1F c1(C(=O)NC2CC(CCC(N)=O)C2)cnn(CCNC(=O)CCOC2CC2)c1 C1(CNC(CCCSC)=O)CCN(C(=O)Cc2cccc(C3CC3)c2)CC1C c1(C(N2CCCC(NC(=O)CCC(F)F)C2)=O)ccc(=O)n(C2CC2)c1 N1(C(C2C(C(=O)NC3CC3)C2)=O)CCc2cc(F)ccc2C1.C1CN1 C(C(C)(O)CC(=O)N(C1CCCN(C(C2CC(O)(CC(C)C)C2)=O)C1)CC)OC C(CCC(C)C(=O)NCC1(C(N)=O)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1)OC N1(C(CC(C=C)(C)C)=O)CCC2CN(C(c3nn(C)cc3SC)=O)CCC2C1 Cc1nnc2sc(C(=O)NCC3CC(F)CN3C(=O)C=CC(C)C)c(N)c2c1C C(=O)(CCC(=O)NC1CC(NC(C2CC3(C2)CC3F)=O)C1)N(C(C)C)C C(=O)(C(F)(F)CO)NCC1C(C(N(CCC(N)=O)CC)=O)CCO1 C1(CCC)CN(C(=O)CC2CCC(O)C2)CC1CN(C(C)CCO)C N1(C(c2cnc(C)n2C)=O)CCC(CO)CC1C(=O)N(C1CC1(C)C)C C1(C2CN(C(=O)CC3(O)CCOC3)C2)(NC(C2CCCOCC2)=O)CC1 N1(C(c2c(CC)onc2)=O)CCC(C2(NC(=O)CC3(C#N)CCC3)CCC2)CC1 C1(NC(C2C=CC(C)(C)CC2)=O)CC(C(N2CCC2C(N)=O)=O)C12CCC2 C(CC(=O)NOCCC(C)O)N(C(COCC(=C)C)=O)CCO Cc1cnccc1C(C)C(N1CC(O)CC1c1ccc(F)cc1)=O C1(C(N2CCC(NC(CC(CC)SC)=O)CC2C)=O)(OC)CCCCCCC1 c1(C(C(=O)N(CC(CN(C(c2cc(CC)on2)=O)C)O)C)(C)F)ccc(F)cc1 C1(C(=O)NCC(CCNC(=O)CN2CC(C)(SC)C2)OC)CC2C(C1)C2(F)F c1(NC2CC(CNC(c3c(CC)onc3)=O)C2)nc2ccc(N)cc2s1 C1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CCCC2)COc2cc(F)ccc2O1 C1(NC(c2nc(C)sc2C)=O)CCCC(C(=O)NCC2CC2(F)F)CC1 C1(NC(COCCCCC)=O)CC2CCC(C1)N2c1ncns1 N1(C(C2(SC)CC2)=O)CCC(C=CC(=O)NC(C)Cc2ncn(C)n2)CC1 N12CCOCC1CC(=O)NCC(CC)(C(CC)(C(C)O)SC)CC2=O c1(C(N(CC(O)CNC(c2cnnc(O)c2)=O)C)=O)ccc(C2CC2)nc1O N1(C(C(CCC)c2ccccc2)=O)CCCN(C(c2cccs2)=O)C(C(C)C)C1 c1(C(=O)NC(CNC(C2N(C(=O)NC)CCC2)=O)C)ccc(C(F)F)cc1 Cc1nc(-c2ccc(Cl)cc2)sc1CNCCC1COC(C)(C)C1 c1(N2CC(CC(C)NC(C3CCSC(C)C3)=O)C2)ncc(C#N)cc1F S(=O)(=O)(c1ccc(C(N2CCCOC(C)C2)=O)c(F)c1)N1CC(C)SCC1 N1(C(C(C)O)=O)CC(O)(C2CCN(C(=O)C=CC3CCCC3)CC2)C1 c1(C(N2CCCC(NC(C(C)C#N)=O)C2)=O)csc2c1CCCCCC2 Cn1ccc(=O)c(C(N2CC(C)(NC(C3CCC(C(F)F)CC3)=O)C2)=O)c1 C(=O)(C(C(C)(C)C)N1CCCC1=O)NCC(CNC(c1c(C)[nH]c(C#N)c1)=O)O N1(C(C(C)=C(C)C)=O)CC2(CCC2NC(C2CCCN2C(c2cccs2)=O)=O)C1 C(=O)(CCCC(F)(F)F)N(C1CCCCN(C(c2ccc(C(F)F)o2)=O)C1)C C(=O)(C(CNC(=O)CCN1CCCCC1)C(C)C)NCC(C#C)C(C)C N1(C(c2ccc(CC(C)C)cc2)=O)CC2(CC2)CC1C(=O)NCc1ncccn1 CCCCCCCC(=O)NCc1cnc(CC)s1 N1(C(C2(C=C)CCC2)=O)CC2CC(NC(C3(CF)CC3)=O)CC2C1 C1(NC(C2(N(C)C)CC2)=O)CC(CNC(=O)C(O)C2CC2)C1 c1(OC)ccc2c(C(=O)Oc3cccc(F)c3O)csc2c1 C(=O)(CCC=C(C)C)N(CCC(=O)N(CCCC)CCCC)C1CCCC1 C1(c2ccccc2)(C(=O)NCC(C(C)C)NC(=O)C(C)(Cl)Cl)CC(F)(F)C1 C1(CC=C)(NC(=O)COC)CCCN(C(=O)CC2(CO)CC2)C1 N1(C(C(C)CC(F)(F)F)=O)CC2CN(C(=O)CCCCNC(N)=O)CC2(C)C1 c1(C(N(CC(O)CNC(=O)CSC(F)(F)F)C)=O)ccc2c(c1)OCC2 C12(C(N(C(C)CSC)CC)=O)CC(CN(C(C3(C#N)CC3C)=O)C1)C2 C(=O)(C1CCc2c[nH]nc21)N(CC(C(C)C)OC)C c1(C(N2C(CNC(COCCC#C)=O)C=CC2)=O)cc(Cl)cc(Cl)c1Cl C1(C(=O)NC(C)(CO)CCF)CCN(C(=O)C(F)OC(F)(F)F)CC1O c1(C(=O)NCC2CC(O)(CNC(CS(N)(=O)=O)=O)C2)ccc([N+](=O)[O-])cc1 Cc1nc2cc(C(=O)NC3CCCCC3NC(=O)CCCS(N)(=O)=O)cnc2s1 O=C(NNc1ccc(C(F)(F)F)cc1)C(C[N+](=O)[O-])C(F)(F)F CC1(C)CCC(c2nc(-c3sccc3S(N)(=O)=O)no2)CC1 O=S1(=O)c2cccnc2N1.C1(CCn2cncn2)CCN2CCCC2C1 C(=O)(C1CCCc2nc[nH]c21)CCC1CCN(C(=O)CC(C2CC2)C2CC2)C1 CN(C1c2ccccc2CCC1O)C(=O)Cc1c[nH]c2cccc(Br)c12 C1(OCCNC(CC=CC)=O)CCN(C(=O)C(F)C2CC2)CC1 Cc1c(Br)ccc(F)c1C(=O)NC(C)CNC(c1cc(F)c(F)cc1N)=O c1(CC)ccc(N)c(C(N2CCCN(C(c3nn(C)nc3Br)=O)CC2)=O)c1 C1(C(=O)NCC(CC)NC(c2snc(O)c2Cl)=O)(CC)CCCCO1 c1(OC)nc(C(=O)NC(C)(CNC(=O)CCC2CC2(F)F)CO)ncc1F CCC(C)(C)C(O)C(=O)N1CCCCC(CNC(C2(N=[N+]=[N-])CC2)=O)C1 C1(C(N2CC(CC)N(C(=O)CCC(C)(C)N(C)C)CC2)=O)CCC(N=[N+]=[N-])CC1 Cc1ccc(C(=O)NC2CC(F)(CNC(=O)CCC3CC3(C)C)C2)cc1CO C1(C(=O)NCC(C)C(C)(F)F)CCN(C(c2cccc[n+]2[O-])=O)CCO1 N1(C(C2CC(CC)OCC2)=O)CCN(C(c2cc(C)[nH]n2)=O)CC(C)C1 C(N=c1[nH]c2ccc(F)cc2o1)C1CC2(CC(NC(C(CC#C)(C)C)=O)C2)C1 C1(C)(C(N2CCC(C)(CNC(C(c3c(C)cccc3)C)=O)C2)=O)COCCOC1 C(=O)(N(CC1CCCCC1(C)C)NS(=O)(=O)Cc1csc(C)c1)OCC CC1=CC(C)C(c2cn(CCCC(=O)NC3CCCC3CF)nn2)CC1 Cc1cc(NC(C2CC(NC(C3CCCC(=O)N3C)=O)C2)=O)cc(C)c1C c1(C(=O)NC(CCCNC(C2C(C(=O)OCC)C2)=O)CO)cc([N+](=O)[O-])cn1C N1(C(C(C)NC(COC)=O)=O)CCC(C2(O)CN(C(=O)CSn3cncn3)C2)CC1 C=CC1(C(=O)NC2CC(NC(=O)C3=COCCO3)C(O)C2)CCCCC1 Cc1cc(C(=O)NC2C3CC2N(C(=O)C=Cc2ccc(Cl)cc2)C3)c(O)nn1 N=c1nc(N2CCC(O)(C(=O)NCC(F)(F)F)C2)c2ccc(C(F)(F)F)cc2[nH]1 N1(C(C=CC=CCC)=O)CC(NC(=O)C(=C2CCCCC2)F)CC(C)C1 c1(C(=O)NC2(C)CCC(NC(c3cnns3)=O)CC2)cnc2ccncc2c1 CCC(C)(C)C(C)CC(=O)N(C(C)CNC(=O)C=Cc1ccco1)C c1(NC2CC3(CN(C(CSCC)=O)C3)C2)cccn2nc(C)nc12 Cn1cc(-n2cccn2)cn1.C12CCN1C(=O)CC1(CC1)NC2=O N1(C(C2CCC(C(C)C)CC2)=O)CCCC(C)(CNC(=O)CCc2ccsc2)C1 S(=O)(=O)(c1cccs1)N.c1(C(C2(CO)CCCC2)=O)ccccc1Cn1cncn1 CC1(C(N2CC(CNC(C3CC4CCC3C4)=O)C2)=O)CCC2(CC1)CC2 N1(C(Cn2c(C(=O)OC)cnc2)=O)C(C)(C)CC(OC)C1(C)C N1(C(C=CCC)=O)CCC(CNC(C2CC3(CCC3)CO2)=O)C(O)C1 c1(C(N2C(CN(C(C3C(CC)C3)=O)C)CCC2)=O)cncc(Cl)c1 c1(OCC)ccc(C(N2CC3(C2)CN(Cc2cc(Cl)cnc2C)C3)=O)cc1Br N1(S(CC(=O)OC)(=O)=O)CC2(CN(C(c3cc(F)ccc3Br)=O)C2)C1 c1(OC)cc(C(=O)NC2CC(NC(=O)CC(C)(C)CN(C)C)C(O)C2)ccc1Cl Cc1ccnc(Cl)c1C(=O)NCC1=CCN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC1 c1(C(=O)NCCC(C)(C)NC(C(C(CC)C)C)=O)cc2c(Cl)nccc2s1 c1(C(=O)OC)ccc(C(N2CCC(NC(=O)Cc3cnsc3)CC2C)=O)cc1C C1(C(N(CCNC(C2(CO)CC(F)(F)C2)=O)CC)=O)CCC2(CCC2)CO1 CC12CCC(C(N3CCCC(C)(NC(=O)CC4CCS(=O)(=O)C4)C3)=O)(CC1)CO2 C(=O)(N1OC2CCC1C2)C1N(Cc2ccc(C)cc2Br)CC2(CC2)C1 C12(C(=O)NC(CCC=C)C)COCC1CN(C1CCNC(=O)CC1)C2 C=CC(C)CC(=O)NCCCN(C(c1cc(C2(C)CC2)c[nH]1)=O)CCC(C)(C)C Cc1nc2nccc(NCCC3CCCN(C(=O)C=CC4CC4)CC3)n2n1 C1(NC(C(CN(C(C2=CCN(C)C2)=O)C)(C)C)=O)CCC2(CCCC2)C1 Cc1cccc2cc(C(N3CC4(CCC4NC(C4CC45CC5)=O)C3)=O)oc12 c1(OCC)nccc(C(=O)N(C2CCC(NC(C3CCCCC3)=O)C2)C)c1F C1(C(=O)NCc2snc(C)n2)CN(C(C2CC(=O)NC2=O)=O)CC12CCC2 C(C(C)(C)CN=c1nc2sccc2c(NC2CC2C2CC2C)[nH]1)OC(C)C C(=O)(C1=CC2CCC1C2)NC(C1CCN(C(=O)CNC(c2ccsc2)=O)CC1)C C1(O)(C(C)C)CCCN(C(=O)C(=O)NCCN2CCS(=O)CC2)C1 C1(C(=O)NCCCN(C(c2nccc(C(F)F)n2)=O)CC)CC12CCCC2 N(C(=NCCc1ccc(Cl)cc1)NC(C)CC(F)(F)F)CCCn1c(C)ncc1 CC(C)C(C)(C)C(=O)N1CCOCC(CNC(c2nscc2Br)=O)C1 c1(NC(C(CC(=C)C)N)=O)ccc2c(c1)C(=O)OCC2 N1(C(c2cn(CC)nn2)=O)CCN(C(=O)C(F)(F)C2CCCC2)CC1COC CCC(C)CCCC(=O)N1CCCC1C(=O)N(C)CC1CCN(C(C)=O)C1 c1(OC)ccccc1C(C(C)NC(=O)CC#N)NC(=O)CC1CC1 N1(C(C(F)=CC)=O)C2CCC1CC(NC(c1ccc(-c3ccncc3)o1)=O)C2 C1(CN(C(CCOCC#C)=O)C)COCCN1C(=O)C(C)NS(C)(=O)=O c1(CCC(=O)N(C)CCNC(C2COCCN2C)=O)cc2ccccc2[nH]1 C12(CNC(Cc3c(C)n(C)nc3)=O)CCC1CCN2C(=O)C1=CCSC1 C1(NC(COCCCC)=O)CN(C(c2ccc(O)nn2)=O)C2(CCC2)C1 N1(C(C(C(C)O)C)=O)CCC2CN(C(C34CCC(CF)(CC3)CC4)=O)CC2CC1 N1(C(COC)=O)CCCC1C(C)(C)NC(C1(C(=O)NC2CC2)CC1)=O Cc1ccn(C)c1C(=O)NC(CNC(c1cnn(C)c1)=O)C1CCC1 C(=O)(CCCCCC(C)O)NCC(CCNC(c1c(C)nc(CC)o1)=O)O C(=O)(CC1=CCN(C(C2CN(C)CCN2C)=O)CC1)N(C)Cc1n(CC)ccn1 CCC(C(=O)NCCC1CC(C)=NO1)N(C(=O)C=C1CCOCC1)C N1(C(c2cccc(C(=O)OC)n2)C(=O)NC(C)(C)C)CC(O)CCC1C c1(C(N2CCCN(C(C(C(C)(C)C)C#N)=O)CC2)=O)cc(Cl)cc2c1OCC2 Cc1oc(C)c(C(=O)NCc2csc(C(N3CCCC3CC3CCC3)=O)c2)c1C C(=O)(CCCCC#N)N1CC(CNC(C(CC)N2CCCC2=O)=O)C(N(C)C)C1 C1(NC(c2ncc(OCC)nc2)=O)CCC2CCN(C(C3C4CC5C(C4)C35)=O)C1C2 c1(CCC(=O)NCCN(C(C(CC#C)O)=O)C(C)C)c(Cl)cccc1Br CON(CCC(=O)NCC(C1CCC1)C1CCC1)C(=O)C(F)(F)C(F)(F)F c1(OC)cc(C(=O)NCC(C)NC(=O)C2=COCCO2)cnc1C(F)(F)F Cc1nc(C)c(C(=O)NC2CCOC(CNC(c3nncs3)=O)C2)nc1C N1(N(C)CC2(C)CNC2)CCN(C(=O)Cc2cc(C3CC3)ncn2)CC1 c1(OC)ccccc1C1C(O)CCN1Cc1ccccc1NS(C)(=O)=O CCCCC(CC1CCCN1C(=O)COC(C)(C)COC)CC C=CCCC(=O)OC1(c2cn(C3CC(C(=O)OC)C3)nn2)CCCC1 c1(C(=O)NC23C(CN(C(C4CCN(C)C4)=O)C2)CC3)c[nH]c2nccc-2c1 c1(CCC(N2CC(COC)CC2(C)C)=O)c(C)[nH]c2ccccc12 N1(C(C(c2ccccc2)OC)=O)CCCC(N(C)C(c2cc(C)co2)=O)C1 CC1CC(CNC(C2(C)CCCN2C(=O)CC2CCN(C)CC2)=O)=NO1 Cc1cccc(CNCC23CC2CN(C(c2c(C)nn(C)c2C)=O)C3)c1Br C(C)(CNC(=O)CN1CCCCC1)(CC(C)C)NC(c1cncc(C)n1)=O c1(OC)cc(-c2ccc(-c3nccn3CCN3CCOCC3)cn2)ccc1C Cc1cc(O)ccc1-c1cn(C(C)C(=O)NC2CC(CF)C2)nn1 Cc1nn(C)c2ncc(C(=O)NC3C(C)CN(C(=O)CC(C)(C)F)CC3C)cc12 c1(C(=O)NCc2cccnc2)ccc(=NCc2ccc(F)cc2Cl)[nH]c1 N1(C(CCN(C(c2ncc(OC)nc2)=O)C)=O)CC(S(C)(=N)=O)C1 c1(C(=O)NC2(CNC(C3COCC(C)O3)=O)CCCCC2)ccnc(F)c1F C1(NC(CSc2cccc(C)c2)=O)CCC12CN(C(C1CCCC3(CC3)C1)=O)C2 N1(C(C(C2CC2)OC)=O)CC=C(CNC(C2CCCC2)=O)CC1 C(C)(N=c1cc(Cl)nc(C)[nH]1)C1CCN(C(CCCc2nc(C)sc2)=O)CC1 C(=O)(C(C)(C)C(F)(F)CC)NCC(CC=C)NC(=O)C(C(C)C)N(C)C C12(NC(C3C(CN)CCCC3)=O)CCCC1NCC2 C1(C(=O)NC(C#C)C(C)C)CCN(C(c2ccc(C)cc2)=O)CC1 C1(NC(CCC(Cn2cc(CNC(N)=O)nn2)(F)F)=O)CC2CCC1CC2(F)F n1(CC)cc(C(=O)NCCC(O)CNC(=O)C(=O)NCC(F)(F)F)c(C2CC2)n1 N1(C(c2cccc(C(C)C)c2F)=O)CCN(C(C2CC2C(F)F)=O)CCC1C c1(C(=O)NCC(C2CCCC2)NC(C(c2cncnc2)C)=O)ccncc1Cl N1(C(=O)OC(C)(C)C)CCC2(COC(CC(=O)NCc3csc4cncn34)C2)C1 N1(C(C2(C(C)C)COC2)=O)CCCC(C(=O)NC23CCC(CC2)C3)CC1 O=C1CCC(CC(N2CCC(F)(C(N3CCC3)=O)C2)=O)CN1.C(CCO)N C1(C(=O)NCc2cc(C(N3CC(NC(=O)NC)C3)=O)on2)CC12CCOCC2 Cc1sc2ccccc2c1C(=O)NCC(C)CN(C(=O)C(=O)NC1CC1)C C1(C(=O)NC(CC)C(N2CCOCC2C(C)O)=O)CCCC1C1CC1 Cc1c(F)ccc(C(=O)Nc2cccc(-c3ccc(CN(C)C)cc3)n2)c1Cl c1(-c2scc(OC)c2)cnc(C(=O)Nc2oncc2C#N)cc1C c1(OC)c(F)cc2nc(NCc3ccc(F)cc3C)sc2n1 Cc1oc(C)c(C(N2CC3CC(NC(c4cc(C(F)(F)F)cs4)=O)C2C3)=O)c1C c1(C(=O)NC2CN(C(C3(C(C)C)CCC3)=O)CC2F)cc(Cl)c(Cl)nc1Cl c1(C(=O)OC)cc(S(=O)(=O)C(N2CCC(CCC(N)=O)CC2)=O)cn(C)c1=O C1(c2c(Cl)ccc(NC(CC)=O)c2)CCCCN1N1C2CCC1CC(=O)NC2 c1(OC)nccc(C)c1C(=O)N(CCn1cc(CCN2CCC(C)CC2)nn1)CC n1(CC(N2CCCC(C)(CNC(=O)CN3CC=CC3)C2)=O)cc(S(C)(=O)=O)cn1 c1(CN(C(C2C3CN(C(C4CN(C)C4)=O)CC23)=O)CC)ccc(C)c(C)c1 c1(C(=O)NCCC(CCNC(C2C(CC(C)C)C2)=O)C)cccc(Cl)c1F C1(CNC(C2(OC)CC2)=O)CCCC12CCN(C(c1n[nH]c(C)c1N)=O)CC2 CC1(C)C(C(F)(F)F)CCN1C(=O)COc1cccc(C#N)c1 C1(O)(c2cc(CN(C)CC3N(C(c4ccn(CC)n4)=O)CCC3)on2)CCOCC1 C1(NC(C(C)NC=O)=O)COC2(C1)CN(C(C13C4C5C1C1C3C4C51C)=O)C2 C1(C(=O)Nc2ccc(-c3ncon3)cc2)CCc2scnc2C1 C1(C(=O)NCCC(C)(C)NC(CCNC(COC)=O)=O)CN2CCC1(C)CC2 CC1CC2CN(C(=O)OC(C)(C)C)CC2N1C(=O)CSc1cc2ccccc2o1 c1(-n2c(Cc3cc(C)sc3C)nc(CC)n2)cc(C)n(CC)c1C C1(C(=O)NCC2CCC(NC(CC3C(OC)CC3)=O)CC2)CC12CCSCC2 C1(CCC)CN(C(c2ccsc2C)=O)CCN1C(c1ccc(Cl)c(OC)c1)=O C(=O)(C(F)C(C)(F)F)N1CCCC(CC(=O)NCC(C)OC(F)F)C1 c1(C(=O)NC(CNC(C(C(CC)O)(C)C)=O)CO)cc(C)c2c(O)n[nH]c2n1 c1(C(C)C)nc(N2CCN(CCCNC(=O)C(C)(C)CN(C)C)CC2)cc(Cl)n1 C(CCCCCC(=O)N1CCOC(C(=O)NC2CC2)C1)SC.C1(C)CCC(=O)N1 CC(C)C(C)(C)C(c1nnnn1C1CC1)NCC1CC1c1ccsc1 c1(C(N2CCCC(N(C(Cc3cccc(CO)c3)=O)C)C2)=O)cnccc1C#N C12(C(=O)OC)CCCC(C(=O)NCCCNC(=O)CC3CCCCCC3)(CC1)C2 c1(CC)ccc(N2CC(C(N3CC(C#N)(CC)C3)=O)CC2=O)cc1 N1(C(c2c(C)cccc2)=O)CC(NC(=O)NC(c2cc(Cl)cc(Br)c2)=O)CC(F)C1 C1(C)(C(=O)NC(c2cc(C)on2)C)CCN(C(c2conc2C)=O)C1 C1(C(N(C)CC2(NC(c3ccn(C(F)F)n3)=O)CC2)=O)CCc2n[nH]cc2C1C c1(C(=O)NC(C2OCCN(C(C(CNC(C)=O)(C)C)=O)C2)C)cnc2n1CCS2 c1(C(CC(=O)NCCCOCCOCCNC2C(C)C2)=O)ccoc1C=O.CO n1(CC(=O)NCC(C)(C(C)C)NC(C(COC)COC)=O)cc(Cl)c(O)nc1=O c1(C(=O)NCC(C(C)(C)C)NC(C(C=C)(C)O)=O)cccc(OC)c1C Cc1oc2ncnc(O)c2c1C(=O)NC1CC1CSc1ccccc1N(C)C C1(CC(=O)NC(CCC)C2CCC2)CN(C(=O)CCC2(C)CC2)CC12CC2 C#CCCC(=O)N1CC(O)(C(F)C(=O)NCCCN2CC=CC2)C1 C1(CC)CCC(F)(CNCc2nc(NC(=O)OC(C)(C)C)no2)CC1 CCC(CC(C)C)C(=O)NCC1CCC2(CN(C(=O)Cn3nnc(=N)[nH]3)C2)O1 C#CCC(C)C(=O)N(C)CCN(C(=O)CN1CCN(c2ccccc2)CC1)C1CC1 C(C)(CO)(C(=O)NCc1ocnc1C(=O)NC1CC(O)C(F)C1)OC c1(OC)ccc2c(CCC(=O)N(CC(C)NC(=O)C#CC3CC3)C)c[nH]c2c1 Cc1cccc(NC(=O)NNC(C)CC#N)c1O C(C(=O)NNc1cc(Cl)ncn1)N1C(C)CCCC1C c1(C(=O)NCC(CO)NC(=O)CCc2cnoc2)cc2n(n1)CCCC2O C(CS(=O)(=O)Cc1ccccc1)NC(N(CC(CC)C)C1CC1)=O C1(C(C)C)(C(=O)NCCCOCCC(=O)NC(C(C)C)c2ccco2)COC1 CN(CCCC(=O)NCC1CC(CNC(c2cncc(O)c2)=O)C1)N=O N1(C(=O)C(Cl)=CCl)CCC(C2CCN(C(=O)CCCc3cccs3)C2)C1 N1(C(CCNC(CC(C)C)C)=O)CCC(C2CC2)(CNC(=O)COC(F)F)C1 CC(CCC(=O)N=c1ccn(CC(N)=O)[nH]1)NC(C1C2CCCCC12)=O CC1OC2(C(=O)NCC3CC(CNC(C4CN(C5COC5)C4)=O)C3)CCC1CC2 C1(C(=O)NCC(C)NC(C(CC(=O)OC)C)=O)CC2CCCCCCC12 CCC(C)(C)C(O)C(=O)N1CCCCCC(NC(c2cccc(C3CC3)c2)=O)C1 c1(N2C(CNC(CCCCSC)=O)CCCC2)nc(Cl)nc2c1CCOC2 C1(N(C(=O)C(C)n2ccnc2)CC)CCN(C(=O)Cn2cnc(=N)[nH]2)C1 Cc1cc(OCC(C2CC2)NC(N2CC(N3CCCCC3=O)C2)=O)cc(C)c1 N1(C(Cn2ccc(C)n2)=O)CCCC(C)(CNC(=O)CCN2CCC(F)C2)C1 Cc1ccc(CNC(C2(C(C)NC(=O)COCC(C)(C)C)CC2)=O)o1 C(CCC(c1nnnn1CCCOC)NC(C)CC1CC1)OCC CC1(C(=O)NCC(c2ccccc2F)NC(C2CCOC2)=O)CC2(CC2)C1 n1(CC)ccnc1C(c1nnnn1C1CC1)NCCOCCC1CC1 CC#CCC(C(=O)NCC(C)Cc1ccco1)NC(c1cncc(OC)n1)=O C=C=C(C)CC(=O)NC(C)CC1CCN(C(c2cccn2CC)=O)CC1 N1(C(C(CC2CC2)OC)=O)CCC(C)(CNC(=O)C(F)CC2CCOC2)CC1 N1(C(C(C)NC(=O)C2CC2)=O)CCC(NC(C2(F)CCOC2)=O)C2(CCC2)C1 C1(C(N2CC(C)(NC(C(CC)NC(C)=O)=O)C2)=O)COc2ccc(F)cc2C1 c1(C(=O)NCCN(C(=O)Cn2cc(C(C)O)nn2)CC)coc(C2CCC2)n1 c1(CNC(C(C)SCCCC)=O)cccc(C(=O)NCc2cncn2C2CC2)n1 c1(C(N(CC(C)NC(C2(O)COC2)=O)C)=O)cc2cc(Br)sc2s1 Cc1ncc(C(=O)NC2CCC(CCNC(C3(O)COC3)=O)C2)n1C C1(C)(CC)CN(C(c2ccc(C)cc2F)C(=O)NC2CCCC2)CCO1 c1(C(=O)NCCC(C)NC(=O)C(C)CCc2ccccc2F)cnccc1C#N n1(CCCOC)ccc(=NC(=O)CC2(NC(c3cnn(C)c3Cl)=O)CCC2)[nH]1 c1(C(C)NC(=O)Nc2csc(C(C)(C)C)n2)cnn2c1OCCC2 C1(C(C)C)CCCC(OCC2N(C(=O)OC(C)(C)C)CC2(C)C)C1 n1(C(C)C)cc(Br)cc1C(=O)NCC1CC(NC(c2ncccc2N)=O)C1 CC1CCN(C(=O)Cn2cnc([N+](=O)[O-])c2)CC1NC(=O)Cc1c[nH]ccc1=O CC(C)C(CNC(=O)C(c1ccccc1)N(C)C)NC(=O)C(C)S C1(CN(C2CC3CCC2O3)C(C(=O)NC2CCC2)=O)CC(C2CC2)=NO1 N1(C(C(C(C)(C)C)NC(N)=O)=O)CC2(CN(C(=O)CCF)C3CC3)CCC1CC2 N(C(=NCC(C)C)N1CCC(C)C2(CCC2)C1)CC(C1CCC1)OC C1(C(=O)Nc2cccc(C(C)F)c2)CN(C(C2(Br)CC2)=O)CC(C)(C)C1 N1(C(COCC)=O)CCCC2(CCCCC2NC(=O)C(C)Oc2cccnc2)C1 C(C(=O)NC1(C)CN(C(c2cnccc2N(C)C)=O)C1)(C(C)C)CSCC c1(CC(C)NC(=O)C(C2CCCO2)SCC(=O)NCC(C)(C)C)ccc(O)cc1 C1(CNC(c2cn(CC3CC3)nn2)=O)CCC(NC(C2CC2Cl)=O)CC1 N1(C(CC(C=C)CC)=O)CCC2CCC(C1)N2C(C1CCC(=O)N(C2CC2)C1)=O c1(C(=O)NCCNC(C2C(OC)CC(OC)C2)=O)cc2cccc(C)n2n1 c1(C(N2C3CN(C(C(C(C)OC)O)=O)C(CC3)C2)=O)cc(Cl)c2c(c1)OCCO2 c1(C(C)=O)ccc(C(=O)NCc2cc[nH]c2C(=O)NC(C)C2CC2)[nH]1 c1(C(=O)NC2CCCN(C(=O)CO)CC2)ccc2nncn2c1 N1(C(C(CC)OC)=O)CCc2ccccc2C(NC(=O)C(O)c2ccsc2)C1 c1(NC(C(N2CC3C(NC(C4CCC(CC)O4)=O)(C3)C2)=O)=O)c(C)cccc1C c1(N(C)C)cc(C(=O)NC2CCCC(CNC(=O)C3=NOCC3)C2)ccn1 CC(C(C)(C)C(=O)NOCCC1CC1)NC(c1ccn(C)c1)=O C1(CC)CN(C(C2CCC2)=O)CCC1NC(=O)C(O)Cc1ccccc1 c1(CC(=O)N(C2CCC(NC(=O)C(F)(F)CO)C2)C)cccc2c1OCCO2 c1(OC)ccc(S(=O)(=O)N2CCCC(NC(c3cccc(C(F)F)c3)=O)C2)cc1 CCCCC(C(=O)NCC(C(N1CC2CC1(COC)C2)=O)N(C)C)C(C)C C(=O)(C#Cc1ccccc1Cl)OCc1c(S(C)(=O)=O)cccc1 C=CCC(C)(CC)C(=O)N1CCOCC1CN(C)C(C1CCOC2(CCC2)C1)=O CCCCC(C(=O)N1CCC(NC(=O)Cc2sc(S)nc2C)C1(C)C)N(C)C c1(CN(CC(C)C)CC2CCCO2)cnc(-c2cccs2)s1 CC1(C)CC(NC(c2cnnc(O)c2)=O)CCN(C(=O)C=Cc2ccncc2)C1 C1(C(=O)NC2C=CC(C(=O)OC)C2)CCCCN(C(=O)CC=C(C)C)C1 C(=O)(C(C)C(=O)NCC1CC(C(=O)NCC#CCCO)CO1)OC C#CCCC(C(=O)NC(CC1CC1)C(=O)NC)NC(c1ccc(O)c(C)c1)=O C1(NC(C)=O)CC(C(C2CC2)NC(=O)C(C)Oc2ccc(F)cc2Cl)C12CCC2 CCCCC(C(=O)N(CCNC(=O)Cc1nc2c([nH]1)CCCC2)CC)C(C)C CC(C)P(=O)(CC(=O)NCC#CCNC(C1CCS(=O)(=O)C1)=O)C(C)C N1(C(c2cnn(C3CC3)c2)=O)CCCCCC1CNC(C1CC(F)(CO)C1)=O c1(OCC)ccc(N=c2scc(-c3cnn(C)c3)n2-c2ccco2)cc1 c1(C(=O)NC2CC(NC(c3c(OC)cccc3)=O)C2)cccc2nonc12 Cc1cscc1C(N1CC(O)(C(C)NC(c2cc(-c3ccco3)[nH]n2)=O)C1)=O c1(OC)cc(C)c(C(=O)NC2C3CCC(C3)N2C(=O)CCCOC(C)C)cn1 c1(OC2CC(NC(CC(C)(O)c3ccccc3)=O)C2)cccc2c1CCS2(=O)=O C(=O)(C1CCCc2cccnc21)N1CC2CN(C(C(CC)(C)CO)=O)CC(C1)O2 c1(OC)ccc(C(N2CCC(NCc3cc(Br)ccc3OC)C2)=O)c(OC)c1C N1(C(c2c(CC)cns2)=O)CC2(C1)CN(C(c1scnc1CC)=O)C2 N1(C(C2(C)CCOC2)=O)CCOC(C(=O)NCC(c2ccco2)O)CC1 CN1CCc2ccc(C(=O)NCCC3(NC(=O)CC(C)(C)C4CC4)CCC3)cc21 N1(C(c2cccc(C)n2)=O)CCC(C)C(N(C(=O)COCC(C)C)C)C1 Cc1ncc(C(=O)NCC2=NOCC2)c(Br)c1Cl C1(C(N(CCCC)CCCO)=O)CN(C(=O)C2=CCCC2C)CC1(C)C C(=O)(C1=CCN(C(=O)C(C)CN(C)C)C1)NCCCN1C(C)CCC1 C(C(C)CC(=O)NCC1CCCC1NC(c1c[nH]nc1Br)=O)OC C12(C(=O)NCC(CC(=O)OC)O)CCC(CC1)N(C(=O)C(C)N(C)C)C2 C1(C(=O)NCCC2CCCN(C(=O)CC(F)(F)Cl)C2)(OC)Cc2ccccc2C1 Cc1cc(C(=O)NC2C3CC4C2C4C3C(N2CCC(O)(C(C)C)C2)=O)cnc1C C(=O)(C(F)C(F)(F)F)NC(CN(C(C1OCCC1C(C)C)=O)CC)C N1(C(CCC(N)=O)=O)CC(CNC(c2nscc2Br)=O)C2(CC2)C1 c1(CC(=O)NC(C)CN(C)C(c2csc(Cl)n2)=O)ccn2cncc2c1 Cc1ccc2c(c1)CN(C(c1cccc(NCc3cccc(O)c3F)c1)=O)CC2 c1(CNC2CCN(C(CC(=O)OCC)=O)C2)ccn2ccnc2c1 C1(NC(CC=CC)=O)CN(C(=O)CCc2cnc[nH]2)CCC1CO Cc1cc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)C2CCC2)c(F)cc1Cl CC1(C)C(NC(=O)Cc2ccsn2)C2CCCN(C(=O)CC3CCCCCC3)C12 CN1CC2C(C(=O)NC3CC(NC(=O)CCN(c4ccncc4)C)C3)C2C1 C1(CCC)CCC(C(N2CCCC2CCNC(C2CC2CCC)=O)=O)CC1 C1(NC(CC(C)CF)=O)CN(C(=O)CCc2ccc(Cl)nc2)CC1(C)C C1(NC(c2nnn(C(C)(C)C)n2)=O)CC2CCC1N2C(c1cc[nH]n1)=O c1(C(N(CCCC)C)=O)ccc(C(F)(F)F)cc1-c1ccc(-c2cccnc2)s1 N1(C(C2(CC)N(C(C(=O)OCC)=O)CCC2)=O)CCC(C#CC)C1 CCCCC(CC)C(=O)NC(Cc1cc[nH]n1)C(=O)NCC1CC1c1cccnc1 c1(C(=O)OC(C(=O)NC(COCC)(C)C)C(C)C)ccc2c(c1)OCO2 CCCCC(C)C(=O)N1CCCC1(C(=O)NCc1n[nH]c(C)n1)C(C)C CC(C)(CNC(=NCC1CC1)NCc1nnnn1C1CC1)C(F)(F)F CCC(C)C(=O)N1C2CCN(C2)C(=O)C1.C(=O)(C(O)CSC)N c12nc3sc(C)cn3c1C(=O)NCCNC2=O.C(O)(C(F)(F)F)C1(CC)CCC1 C1(CNC(=O)NC(c2cccc(F)c2F)C)COc2ccccc2O1 N1(C(CC(=C)C)=O)CCCCC1CCN(C)C(c1ccc(NC(C)C)cc1)=O CCC(CNC(=O)C(F)Cc1ccccc1)(CC)NC(=O)CN1CSCC1=O O=C(C1=C(Cl)CC1)NC1CCC(NC(=O)CCSCc2ccccc2)CC1 S(=O)(=O)(c1ccc(Cl)cc1)CNC1(CCCNC(=O)OC(C)(C)C)CC1 c1(CN(C(c2cc(C)ns2)C(=O)NC2COC2)C)ccc2c(c1)C(=O)N(C)C2=O c1(C(=O)NC23CC(NC(C4C(C)SCCC4)=O)(C2)C3)c(Cl)nc2ccccn12 C(=O)(C1CCCn2ccnc21)NC1CN(C(c2ccnc(C)c2C)=O)CC1C C=C(C)CC(C(=O)N1CCC(O)C1C(=O)N(C1COCC1O)C)OC c1(C(=O)OC)cnc(C)[nH]c1=NC(C)CNC(C1CC2CCC(C1)C2)=O C(=O)(CC(O)CCSC)N1CCC(CC(C)NC(CC=CCC)=O)CC1 N1(C(C2C(C(C)C)(CC)C2)=O)CCCN(C(c2ccc(C)cc2)=O)CCC1 C(CCCC)(C(=O)NC(C)CCCC)NC(CC=CC=C)=O C(=O)(CCN=C(NCc1cccc(OC)c1C)NC(C)C(F)(F)F)NC c1(OC)ccccc1NCC(=O)NC1CCC(NC(=O)C(C2CCC2)OC)CC1 N1(C(CC(=O)OC)=O)CCCC2(CCC(NC(=O)Cc3cn(C)cn3)C2)C1 C(CN=[N+]=[N-])(C(=O)N(C)CCn1ccnc1)NC(c1n[nH]c(C)c1C)=O C1(C(C)(C)O)CC(NC(=O)CC2CC(NC(C3CCSC3)=O)C2)C1 c1(C(C(N2CCC(NC(C3C(OC)CCC3)=O)CC2)=O)(F)F)ccc(F)cc1C C#CC1(C(=O)NC2CCN(CCCO)C2)CN(C(=O)COCC(C)(C)C)C1 Cc1nc2c([nH]1)C(C(=O)N1CCN(C(=O)CC3CCC3)CC1CC1CC1)CCC2 C1(C(N2C(C(N)=O)CC2)=O)CC2(CC(N(C(C3CC4(CCC4)C3)=O)CCO)C2)C1 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCCCN1C(C1CCCOC1)=O C(N=c1[nH]cnc(NCC(=O)NC(C)(C)C)c1C)C1(OC)CCCOC1 c1(C(=O)NCC(CN(C)C(C2CNC(=O)N2)=O)O)cc2n(c1)CCSC2 C1(O)(CNC(=O)CS(=O)(=O)NC(C2CCC(CC#N)CC2)=O)CCN(C(C)=O)C1 c1(CC)ccc(C(=O)NC(C)CCNC(=O)Cc2cc(C)no2)s1 N1(c2[nH]c(N(c3ccccc3)C)nc(=NC)n2)CC2(C)CN(C)CC2(C)C1 Cc1csc(C(c2nnnn2C2CCOC2)NCCCC2CCC2)n1 c1(C(=O)OCC)cccc2c(CO)[nH]nc12.N12CC3CCCN3CC1C2=O c1(NC(C(N(OC)Cc2ccc(C)o2)=O)=O)ccccc1S(=O)(=O)C(F)F N1(C(C2CC(C)(CNC(CCSC)=O)C2)=O)CC(C)C(C)C1C CON(CCC(=O)N1CCOC2(CCC2)C1)C(=O)C1OCC2CCCC12 c1(OC)ccncc1CNC(C1(C(C)NC(C2CCC(=O)C2)=O)CC1)=O c1(OC)cnc(NC(=O)NC(c2nccn2C)C(C)C)nc1 c1(OC)cccc(CN(C(=O)C(C)(C2CCC2)NC(c2cccc(OC)c2)=O)C)c1 C1(C(N(CC#C)CCF)=O)CCOC1COC1CN(C(=O)CCOC)C1 Cc1csc2ncnc(NC3CN(C(C45CCCC(C4)OC5)=O)CC3C)c12 CC(CC(=O)NCc1ccc(-c2ccc(SC(F)(F)F)cc2)nc1)CC(C)(C)C C=CC1CN(C(c2ccc(C(N)=O)cc2)=O)CC1NC(=O)CC1CC1(C)C c1(OC)ccc(S(=O)(=O)NC2COC3CN(C(=O)Cc4cncnc4)CC23)cc1 N1(C(C(C)C)=O)CCCCC1C(=O)OC(C)C(N1CCOCC1)=O c1(C(=O)NC(C(=O)N(C(CC)C2CC2)C)CC2CCCC2)cc(C)c(F)cn1 N1(C(CCC(=C)C)=O)Cc2ccnn2CC(NC(=O)C(C)OC2CCCCC2)C1 C(Cn1cncn1)(C(=O)NCc1c[nH]nc1C1CC1)NC(c1ccon1)=O C(=O)(C(CC(F)F)C1CCC1)N1CC(NC(CCOC(C)C)=O)C(C)C1 CC1(C#CC(=O)NC(C)(C)C(N2CC3CC(N4CCCC4)C2C3)=O)COC1 Cc1cc(C(=O)NC(CNC(c2cc3[nH]ccc3s2)=O)C(C)(C)C)cc(C)c1F C1(CCC=C)(CNC(c2ccc(CC#N)s2)=O)CCCC1 c1(C(=O)NC2(C)CCCCCC2)ccc2nnc(C3CC3)n2c1 S(=O)(=O)(c1cc(F)ccc1C)NC1C(OC)CN(C(=O)C(=O)NCCN(C)C)C1 C(=O)(C(O)CCC1CC1)N(CCN(C(=O)C(C)(C)c1cncnc1)C(C)C)C CON=CC(=O)NC(c1cnn(C)c1)C(=O)NCCn1cnnn1 c1(C(N(CC(C)NC(c2c(C)ncs2)=O)C)=O)ccc(OC(C)C(F)(F)F)nn1 C1(CNC(CCn2c(C)ncc2)=O)CC2CCC(C1)N2C(=O)Cn1[nH]cnc1=N c1(C(C)C)ccc(C(N2CCCCC(NC(=O)C=Cc3ncco3)C2)=O)c(F)c1 N1(CCNC(c2cncc(Cl)n2)=O)CC2CC(C(F)(F)F)CC1C2 C(N=c1[nH]c(=NCc2ccc(Br)o2)[nH]c2c1CSC2)c1cc2c(s1)CN(C)CC2 c1(CNC(C(c2ccccc2)NC(COC(CC)CC)=O)=O)csc(O)n1 c1(CN(C(CN(C2CCC2)C(C)=O)=O)C)noc(C2CC2)n1 c1(C(=O)NCCCNC(C2CCC(N(C)C)C2)=O)cccc2c1CCOC2 CC(CC(F)(F)F)C(=O)NC1CCCN(C(c2nccc(C(F)F)n2)=O)C1 c1(C(=O)NCC(C)NC(c2ccoc2)=O)nc2c(Br)cncc2[nH]1 C(=O)(C1=Cc2ccccc2C1)c1nnc(N2Cc3c(nc(C)s3)CC2)n1C C12(NC(C(C)NC(N)=O)=O)CCOC(CNC(c3nc(Cl)ccc3N)=O)(C1)C2 CC(C)CC(O)C(=O)NCCCCNC(=O)CC(C(F)F)N1CCOCC1 N1(C(C(CCCOC)NC(c2cc[nH]n2)=O)=O)CCOCC2(CCC2)C1 c1(C(N2CC(CC(C)NC(CSCC)=O)C2)=O)cc(C)[nH]c(=NC)n1 N1(C(C2C(C=C)C2)=O)CCN(C(=O)CCOC2CC2)CC1c1ccnn1C C(=O)(CCC(C)C)NCc1ccc(CNC(c2c(CCC)[nH]cc2)=O)s1 C(c1ccc2c(c1)OCO2)=CC(=O)NC(C)CNC(C1CS(=O)(=O)CC12CC2)=O C(C(F)(F)CC(=O)OC)N(c1cc(NC2CC2)ncn1)Cc1c(OCC)cccc1 N#Cc1ccc(C(=O)NCC(=O)NCC2CC2NC(=O)C2=NOCC2)cc1 Cc1ccc(F)c(C(N2CCC(O)(CC(=O)NCC3CC(=C4CCC4)C3)C2)=O)c1 c1(C(=O)NC(CC=C)CNC(=O)Cc2ccc(C)nc2)nn(C)c(C)c1Cl C1(C(=O)NCC2CC(C(N3C(CSC)CCC3)=O)C2)CC(F)CN1C C(=O)(C1=CC(O)CCC1)NCC1(F)CCC(CNC(=O)CCc2cccnc2)C1 c1(CC)nc(C(N2CCC(NC(=O)CC3CC3(Cl)Cl)CC2)=O)c(N)s1 CC1CCN(C(=O)CN(C2CCCC2)C)CCN1C(=O)Cn1cccn1 C(=O)(C(C)N(OC)C(=O)CCCNC(=O)CCCCN(C)C)OC c1(C(C)=O)ccc(C(=O)NC(C)CNC(C2CC2C)=O)[nH]1 CC1(NC(c2ccc(C(N)=O)s2)=O)CCN(C(=O)C(C)(C)C2CCC2)C1 C1(C(=O)NCC2(C(N)=O)CN(C(CCNC(=O)NC)=O)C2)CCCOCC1 N1(C(=O)Cc2ncccc2F)CCCCC(CO)C1.C1(C2CCOC2)C(=O)N1 C(C1CCN(C(c2cccc(Cl)c2)=O)CC1)=CC(=O)NC(CCSCC)C C(=O)(CC(C)C(C)C(C)C)N1CCC(CN(C(c2cc(C)cc(Cl)c2)=O)C)CC1 CS(C)(=O)=Nc1cccc(C(N2CCCCC2Cc2cccc(Cl)c2)=O)c1 N1(C(c2oc(CC)c(C)c2)=O)CCCN(C(C2CC(C)(C)CO2)=O)C(C)C1 c1(C(=O)NC2CCC(C(F)(F)F)C2I)cnc(-c2nn[nH]n2)c(Br)c1 Cc1ccnn1C(C)C(=O)N(C)CCOCCNC(=O)CCCC1CC1 N1(C(CCNC(COC)=O)=O)CCCC12CCN(C=O)C2.C1(CC(C)C)CN(C(C)=O)C1 C1(n2cc(COCC)nn2)CCCN(C(=O)CC(=O)Nc2cccc(F)c2)C1 c1(CCC)sc(C(=O)NCC2(NC(C3CCCC(CCC)C3)=O)CC2)cc1CC C1(NC(C2CCCN2C(=O)CC2CC3(CCC3)C2)=O)C2CCCOC12 C1(C(=O)N(CC(=O)NC(CCO)C2CCC2)C)(CC)CCCCO1 C(CCS(C)=O)(C(=O)NC(CNC(=O)Cc1csnn1)CC(F)(F)F)N(C)C CC(C)(CCCCNC(=O)C#CC1CC1)NC(c1coc(O)n1)=O Cc1cc(N)c(C)nc1C(N1CCC(NC(C2CCN(C)C2)=O)C(O)C1)=O C#CC1(C)CCCN(C(=O)COc2ccccc2C(N)=O)C1 C1(NC(c2nc(COC)oc2)=O)CC2CCC(C1)N2C(c1oc(C)nc1C)=O C1(SC)CCCC(c2cn(CC(F)CCNC(c3ccc(=O)oc3)=O)nn2)C1 Cc1cc(Br)cc2cc(CN3CCC(N(C)C)C3)oc12 N1(C(CCCCC(C)=O)=O)CCCC2NC(=O)CC12 Cc1conc1C(=O)NCCOCCCNC(=O)C(c1ccnn1C)C c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CCCC2)cc(Cl)cc(F)c1N c1(OC)cnc(Cl)cc1C(=O)NCCC(F)(F)CCNC(=O)C(C1CC1)C1CC1 N1(C(c2c(CC)nc(C)[nH]2)=O)CC(C)N(C(=O)C(F)CC(C)(C)C)CC1C N1(C(=O)CCN2CCC(F)C2)CCC2(CCN(C(c3ccno3)=O)C2)C1 c1(OCC)ccc(C(=O)NCC2CC(NC(=O)C3CC3)C(O)C2)cc1C C1(C(=O)NC(CN(C(C2C(C=C)CC2)=O)C)(C)C)CC12CCCc1ccccc12 c1(OC)cccc2c1OCC(C(=O)NC1CC1CNC(=O)C(C(C)C)N(C)C)=C2 Cc1c(C(=O)NC2CCC2NC(c2ccsc2)=O)cnc2c(Cl)cccc12 CC(C)C(CN(C)C)C(=O)N1CCN(C(c2cnn(C(C)C)c2)=O)CC1C1CC1 C1(NC(C(C)C2(C)CC2)=O)CCC2(CC1)CC2NC(=O)CCOC1CCC1 Cc1nn(C(F)F)c(C)c1CC(N1CCC2C(NC(=O)CN(C)CCO)CC12)=O CCC(C(=O)N(CCCNC(=O)Cc1nncn1C)C)N(C)C Cc1cccn2cc(CC(=O)NCC34CC3CN(C(c3ncn(C)n3)=O)C4)nc12 C1(N=c2nc([N+](=O)[O-])[nH][nH]2)(NC(=O)OC(C)(C)C)CC2(CC2)C1 C(=O)(C1CCCc2scnc21)NC(CNC(c1cnc(C)s1)=O)CC(C)C N1(C(C(C)N(C(C2(OCC)CCCO2)=O)C2CC2)=O)CCCC(C)C1 c1(CNC(CN(c2ccccc2)CC(C)C)=O)cc2cc(Br)ccc2o1 Cc1sc2cc(F)ccc2c1CCNC(CCS(=O)Cc1ccccc1)=O C(=O)(C(C)(C)CCCNC(c1cc2cccn2cn1)=O)N1C(COC)C=CC1 C(=O)(C(C(C)(C)C)NC(C1CC(C)(C)CN1C)=O)N(CCC(F)(F)CO)C c1(C(=O)NC(C(C(C)C)NC(=O)CN2CCCCC2)C)ccc2nccnc2n1 CCCC(CCC)C(=O)NCC(O)CNC(c1ccncc1N1CCCC1)=O c1(CNC(NC2C(F)(F)C2)=NCC2CCCCC2)ccc(F)cc1F C1(OC)CCCCN(C(=O)CC(O)CNC2CC(NC(=O)OC(C)(C)C)C2)C1=O CC1CN(C(N2CCN(C)CC2c2ccccc2)=O)CCN1C(=O)OC(C)(C)C Cc1nc(N2CC(NC(=O)Cc3ccc(F)cc3)C(F)C2)c2cc(Br)ccc2n1 CN1C(=O)CCCC1C(=O)N(C1CC(C(=O)NC2CCCC(C)(C)C2)C1)C C(=O)(C1=CC2CC=CCC12)NC1(CC=C)CN(C(C2CCS(=O)(=O)CC2)=O)C1 c1(C(=O)OC)cc(NC2(CNC(=O)CC3CCC(C)CC3)CCCCC2)ncn1 Cc1oc(S(N)(=O)=O)cc1C(N1CCC(C(C)NC(=O)CCNC(N)=O)C1)=O C1(C(N2C(C)(C(=O)NC3C=CC(C(=O)OC)C3)CCC2)=O)CCOCC1(C)C Cc1nc(C)n(CC(N2CCCC2C2(NC(=O)Cc3n[nH]c(C)n3)CC2)=O)n1 N1(C(c2cccc(CC)c2)=O)CCC(CNC(=O)C(C2CC2)N(C)C)CC1C N1(C(c2ccc(S(=O)(=O)NC(CC)C)cc2)=O)Cc2ccccc2C12CCOCC2 C1(NC(CC2C(C)CCO2)=O)CCCC2CN(c3cc(Cl)nc(C4CC4)n3)CC12 C1(C(=O)NC2(CNC(CC(C)CN(C)C)=O)CC2)CCc2cnn(C)c2C1 N1(C(C(C2(O)CN(C(c3ccc(C)nc3)=O)C2)F)=O)CCC2(CCC2)C(O)C1 c1(N(C(c2snnc2-c2ccccc2)=O)Cc2ccccc2)cnoc1C1CC1 C(N=c1[nH]c(N2CCN(C3CC3)CC2)nc(=N)[nH]1)c1cccc(N(C)CC)c1 c1(C(=O)NCC2COCCO2)cnc2n[nH]c(-c3ccc(F)c(F)c3)c2c1 c12cccc(c1Cl)OC2.C(C(=O)N(C)C)SCCOCC N#Cc1cc(S(=O)(=O)N2CC3C(C2C(=O)NC2CCC2)C3CO)ccc1F c1(C(=O)OC)ccc(NCCCNC(c2cncn2C)=O)nc1 N1(C(CC)C(=O)NCC(CC)NC(C2(C(C)C)COC2)=O)CCc2ccccc21 N1(C(c2[nH]cc(C)c2C)=O)CC2CCC(C1)N(C(=O)C(O)C1CCC1)C2 N1(C(c2nc(OC)nc(O)c2)=O)CC2CC1CN(C(C1CCOC(C)C1)=O)C2 C1(C(=O)NCCCN(C(C(CC#C)C)=O)C(C)C)CCC2(CC1)CC(O)C2 c1(CNC(C2(C)CCN(C)C2)=O)cc2n(n1)CCN(C(=O)CC1CCCOC1)C2 N1(C(c2nc(C)nn2C)=O)CCC2CN(C(c3sc(CO)nc3C)=O)CCC2C1 CC(=O)C(C)CC(C)C(=O)NC1(C(=O)NCCN=S(C)(C)=O)CC1 c1(C(=O)NC(CNC(C(CC)O)=O)C2CC2)cccc(C(C)C)c1OC N1(C(c2c(C(C)=O)ccs2)=O)CCN(C(c2noc(C3CC3)c2C)=O)C(CF)C1 CCC(C)CC(C(=O)NCCC(=O)N1CCCC1)NC(c1nnccc1C)=O C1(CNC(CN2CC(CC)C2)=O)CN(C(=O)C(C)CC(N)=O)CC1(C)C N1(C(=O)C2=CCC(F)(F)CC2)CCC2C(CCCN2C(=O)Cc2csc(Cl)c2)C1 N#Cc1ccc(CCCNC(C2C(NC(C3CCCCC3)=O)CCCC2)=O)nc1 C1(O)(CNC(c2[nH]c(=NC)sc2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 C1(C(=O)Oc2ccccc2)COC(C)(C)CN1CCNc1c(C)cccc1 C12(CNC(=O)Cc3ncccn3)CC(CO1)N(C(=O)COCCF)C2 C#CC1(O)CC(C(=O)N(CC(C)CNC(=O)CCn2ncn(C)c2=O)C)C1 c1(CC)cc(NC(=O)C(Cn2cncn2)NC(=O)CC#N)ccc1F c1(C(C)(C)C)c[nH]cc1C(=O)NC1CCN(Cc2cn(C3C=CCCC3)nn2)C1 N1(C(COCC(=C)C)=O)CCN(C(c2snnc2C)=O)C2CCCCC2C1 N1(C(c2ccccc2C(N)=O)=O)CCC(NC(=O)Cc2cccc(O)c2)CC1C c1(NC(c2ccnn2Cc2ccccc2)CC)c(F)ccc(Br)c1F C1(NC(c2n(CC)ncn2)=O)CCN(C(c2ccc(C#N)s2)=O)CC1F C(C)(CCCCNC(=O)CCN1CCCC1=O)NC(C(C)Cc1ccccc1)=O CCCC(C(=O)N1CCCC1C(C)NC(c1cc(C(N)=O)[nH]n1)=O)S(N)(=O)=O C(C1=CCN(C(c2scnc2C)=O)CC1)NC(C(CCSC)O)=O C1(CC(=O)NCCC2(CC3CCC3)CC2)CCN(C(C2CCCOC2)=O)CC1 N#Cc1ccc(C(N2CC(CNC(=O)C=C3CC3)C2)=O)cc1Cl C(=O)(C(C)CC(=O)N(CC(O)CN(C)C(c1ccc(C)[nH]1)=O)C)OC C1(CNC(=O)C=CCN2CCCC2)(NC(=O)CC2COC(=O)C2)CCOC1 N1(C(C2CCCC2Cn2cc(-c3ncccc3Cl)nn2)=O)CCC(CN)CC1 N1(C(C2CC3CC2C3)=O)CCC(O)C(O)C1 CCCC(CCC)CC(=O)NCC(c1ccccc1F)NC(=O)C(C)(CC)CO CC(CNCC#CCOC1CCOC1)CC(F)F C1(C(=O)NCCCN(C(C(F)=CC)=O)CCO)C(c2ccncc2)C1(C)C c1(OC)cc(C(=O)NCCC2(NC(=O)C=C3CCCCC3)CC2)cc(F)c1 C1(C(=O)NCC(CCNC(C2(C)CS(=O)(=O)C2)=O)O)COc2cc(F)ccc2O1 C1(F)(CNC(c2ccc(Br)o2)=O)CC(NC(C2CC(CCF)C2)=O)C1 N1(C(COCCCC#C)=O)CC(O)CC1(C)C(=O)N(C1CCCC1C)C c1(C(=O)NCC2(O)CN(C(C3(C)COC3)=O)C2)ccc2scc(Br)c2c1 CC1(NC(=O)CC2CCCOC2)CCN(CC2COCCO2)CC1 CC1(O)CCCN(C(=O)C(O)C2CN(C(=O)CC3CCCC4CC34)C2)CC1 N1(C(c2nc(C(F)(F)F)nn2C)C(=O)NCCOC)CCOCC12CCSC2 CC1CN(C(C23CCC(NC(=O)C4=NOCC4)(CC2)C3)=O)CCC1=O C1(C(N2C(C)CN(C(c3nc(C(F)(F)F)cs3)=O)CC2)=O)CC2CC1CC2(F)F C1(C(=O)NCC(C2CC2)OC)CC2CN(C(=O)CCCSC)CC2C1 CCC(F)(F)CC(=O)NCC(C1CCCCN1C(=O)C(O)Cc1cnc[nH]1)(C)C O=C(CCC(=O)C1CCOCC1)Nc1ccc(OCCF)cc1 c1(SC)ccc(C(=O)NC(C)C(C)NC(c2sc(-c3ncc[nH]3)nc2C)=O)cc1 C12(C(=O)NCC3C(C)(C)OCC3)CC(CO1)N(C(C1(C)CC=CCC1)=O)C2 C(=O)(C(CCC1CC1)NC(c1coc(C(C)C)n1)=O)NCCCN(CC)CC.CN Cc1nn(C)cc1CCC(=O)N(C(CNC(=O)C(c1ccc(Cl)s1)C)C1CC1)C N1(C(c2c(C#C)c[nH]n2)=O)CC(C)N(C(=O)CCCS(N)(=O)=O)CC1C C=CCC(CC(C)C)C(=O)NCC=CCC(N1CCOCC(C)(C)C1)=O Cn1cc2c(n1)CC(C(=O)NCCCCNC(=O)C1=CC(C)(C)C1)CC2 C1(C)(C(=O)OC)CCN1C(C1CC(C)N1C(C1(COC)COC1)=O)=O C1(NC(c2cnc(-c3ccoc3)s2)=O)CCN(Cc2ncc(Cl)s2)CC1F c1(C(N2C(CNC(CC3CC(COC)C3)=O)CC2)=O)cccc2c1OC(F)(F)O2 C1(C(=O)NCCCN(CCC)C(c2cc(OC)c(F)cn2)=O)CC2(C1)CC21CC1 c1(NC(C2CCN(C(c3cnc(O)cc3O)=O)C2)=O)ccc(Cl)nc1Br Cc1cc(C=CC(=O)NCC(C2CCC2)NC(=O)CCC2CCN(C)CC2)on1 c1(C(C)(F)F)ccccc1NC(c1ccc(C2CC2)cc1)=O CN1CCOCC1C(=O)NC1C=CCN(C(=O)CCNC(C2CCOCC2)=O)C1 N1(C(COC2(C)CCCC2)=O)CCN(C(c2cc(N)ccc2Cl)=O)CC(O)C1 c1(CN(C)C(c2ccc(N(C)C)nc2)=O)cc(S(=O)(=O)N(C)C)cn1C C1(CC#C)CCN(C(=O)C(CNC(=O)C(C)N(C(N)=O)CC)N(C)C)C1 c1(C(=O)NCC2CC(NC(c3cc4scnc4[nH]3)=O)C2)c[nH]c2cccc(F)c12 Clc1ccc(Br)c2c1C(NCc1nccn3cc(Cl)cc13)CC2 C#Cc1ccc(CC(N2CC(NC(C3(C=C)CCCC3)=O)CC(F)C2)=O)cc1 N1(C(CC2(C=C)CCOCC2)=O)CCOCC(F)(CNC(=O)C=CC(C)C)C1 N1(C(c2c(C(C)=O)c[nH]c2C)=O)CC(OC)CC(NC(=O)C(C)CC2CC2)C1 CC1=C(C(=O)NCC(C)NC(c2cccc(-n3cnnn3)c2)=O)C(C)(C)CCC1 C1(NC(CCCc2onc(C)n2)=O)CCCN(C(=O)Cn2cc(C#N)cn2)CC1 C1(C(N2CCC(n3cnnn3)C2)=O)C(O)CCN1C(=O)CSC(F)F C1(C(=O)NC2(CNC(C(C)C)=O)CC2)CC(=O)N(C2CCCCCC2)C1 c1(CC)c(C)sc(N(C(C(=O)NCC2COCCO2)=O)C)c1C(N)=O N1(C(CC2C(CC)C2)=O)CCC(CO)(CNC(c2ncsc2NC)=O)CC1 C1(C)(C(=O)NCCOCCCNC(C(C)OC(CC)=O)=O)CC2(CCC2)C1 C#Cc1ccc(C(=O)NC2CCC(C)N(C(=O)C=C3CCOCC3)C2)c(F)c1 C1(NC(c2cc(O)nc(O)n2)=O)CC2CC1CN2C(=O)CCN1CCOCC1 CC1CN(C(C2(C)CC2(Cl)Cl)=O)CC1NC(=O)Cn1ccc(C(F)F)n1 N1(C(c2cnc(CC)[nH]2)=O)CCC(C)C1CNC(c1ccccn1)=O Cc1ncc2c(n1)CCC(C(=O)NC1CN(C(c3cc[nH]n3)=O)CC1C(F)F)C2 c1(C(=O)NCC2C(NC(C3(F)C(C)OCC3)=O)CCC2)ccc2[nH]c(=N)[nH]c2c1 c1(CC)c(C(=O)NCC(C)N(C)C(C2OCCC2(C)C)=O)cnn1CC(C)C C1(NC(Cn2nc(C)oc2=O)=O)COC2(CNC(=O)CSC3CCCO3)CC1C2 C(C)(C(=O)N1Cc2ccccc2CO1)N(C(C(C)OCCOC)=O)C c1(OC)cnncc1C(=O)NC1(c2nnnn2C)CC1.c12nnn(C)c1C(=O)N2 C1(C(=O)OC)(C(=O)NCC2CC(NC(=O)C(F)(F)c3csc(=N)[nH]3)C2)CCCO1 n1(CC)ccc(C(=O)NC(C)(CNC(=O)CC2CCC(C)(C)O2)C2CC2)cc1=O C#CC1(C(=O)NC2CC(C)(C)C2)CCN(C(=O)Cc2cnns2)CC1 Cc1cc(Cl)c([N+](=O)[O-])cc1NC(c1ccc2nc(C3CC3)ccc2c1)=O C#Cc1cccc(C(N2CC(NC(=O)CC34CCC(CC3)C4)C3(CC3)C2)=O)c1F C1(O)(C(C)NC(C2(C)CC2Br)=O)CN(C(=O)CCC2(C)CC2)C1 CCCCCCCCC(=O)NCC(C)CC(=O)N1CCOC(C(C)(C)C)C1 c1(C(N2C3CCC(NC(C4C(C)C4)=O)(C3)C2)=O)ccc2ccn(CC(F)F)c2c1 CC(CN(C)C)CC(=O)N1CCCC1CN(C)C(c1ccccn1)=O CC1(C)CCC2(CC1)CC2C(=O)NC1CN(C(=O)C(F)OC(F)(F)F)C1 C(=O)(C1Cc2ccccc21)N1CCCCC(CNC(C2CC(C)(C)OCC2)=O)C1 S(=O)(=O)(c1cc(C)ccc1C)NC1CCCN(C(c2cc(C)[nH]c2)=O)C1 C1(NC(C(CCN(C)C)NC(C(C)NC(=O)NC)=O)=O)CC2CCCC2C1 C1(CNC(C2(SC)CCC2)=O)CCN(C(=O)CSc2nncs2)CC1 C1(CC=C)(NC(=O)CC2CC(CC)C2)CCN(C(c2cc(C)cnc2N)=O)CC1 N1(C(C2OCCN(C)C2)=O)CCC(C(N2CC(C(=O)N(C)C)C2(C)C)=O)C12CCC2 Cc1cc(NC(=O)NC2CC2c2ccc(-c3cccs3)cc2)ncc1Cl C12(NC(CCOCC)=O)CCN(C(c3cnc(C(F)(F)F)c(C)c3)=O)CCC1C2 c1(CC)n[nH]c(CC)c1CC(=O)NC1CCN(C(=O)CC2CCCSC2)CC1 N1(C(CC=C=C)=O)CCC(C(C)C(=O)N(c2ccccc2)CC(C)C)CC1 C1(C(=O)NCCOCCCN(C(C2ON=C(C)C2)=O)C)(CC2CC2)CCN(C)CC1 c1(C(=O)NCC2(F)CC(NC(C3CC(C)C3)=O)C2)sc2cccnc2c1Cl C(C1=NOC2CN(C(=O)C=CC3CC3)CC12)NC(=O)CCc1ccc(Cl)nc1 C1(C(=O)NCC2(NC(c3cnc(C4CC4)s3)=O)CCCCC2)CCC2(CCC2)O1 Cc1cc(C(=O)NCC(c2ccccc2)CN)n2ncc(C#N)c2n1 Cc1nccn1C(C)C(=O)N(C1CN(Cc2nc(C(F)(F)F)cs2)C1)C N1(CCC(=O)NCC2C(NC(CC3CC(OC)C3)=O)CC2)CCOCC1 N1(C(CN(C(C)C)C(c2ccc(CO)o2)=O)=O)CCCCCC1C c1(C(=O)OCC2(COC)CCC2)nn(C)c2c1CN(C(C)=O)CC2 C1(C(N(C2CCCN(C(c3cc(C(C)C)on3)=O)C2)CC)=O)CCCN1C=O c1(C(=O)NC(CC#C)C(=O)NCc2nc(N(C)C)n[nH]2)ccc(C#N)cc1 N1(CC)CCN(CC(=O)N(C)CC2COCCN2C(C2CCCCN2C)=O)CC1 c1(C(CC)(CNC(=O)NCc2cc(Br)c(C)s2)CC)cccc([N+](=O)[O-])c1 C=C1CC2(C1)CC(C(=O)N(CC(C)O)CCNC(=O)C(=O)Nc1ccc(F)cc1)C2 Cc1nc2c(C(=O)NC3CN(C(=O)CC(=O)NCC4CC4)CC3C)ccnc2[nH]1 C(C(=O)N(C)Cc1sccc1C)(C(C)(C)C)NC(C1C(CC)C1)=O N1(C(c2c(OC)csc2)=O)CC(C2(NC(C3CCN(C)CC3)=O)CC2)C1 c1(C(=O)NCCN(C(c2c(SCC)cccn2)=O)C)cc(OC)c(F)cc1N CC(CNC(=O)C=CCN(C(=O)CN1CCCCC1=O)C)C(C)(C)C Cc1cnc(CO)c(C)n1.C12CON(C(=O)C3(CCCN3C)c3cn1nn3)C2 C1(C(N2CC3(CCN(c4nccc(OCC)n4)C3)C2)=O)CCC2CCCCN12 N1(C(C(COC(C)C)NC(C(CC#C)O)=O)=O)CC2CC=CC1C2 C1(NC(C2=C(C)OCCC2)=O)CN(C(c2coc(O)n2)=O)C2(CCOCC2)C1 c1(C(N2CC(O)(C(C)NC(C3CC3c3nc[nH]n3)=O)C2)=O)c(F)ccc(F)c1N C1(C(=O)NCC(CNC(C(C)OC)=O)C)CCCC(F)(F)C1 N1(C(CC(=C)C)=O)CCCC1C1CCCCN1C(=O)C1=C(C)CCCC1 NC1CC2CCCC(C1)N2C(=O)C(=O)NC1CC(=O)N(c2ccccc2)C1 c1(C(=O)NC2CCN(C(C(CCCC)NC(N)=O)=O)C2)cc(OC)cc(Cl)c1F c1(OC)cc(F)c(C(c2nnnn2C2CCC2)NCc2sncc2Br)cc1Cl C1(CNC(C(C=C)c2ccccc2)=O)CC2CCC1N2C(c1[nH]nnc1C)=O C1(C(=O)NCC2=CCN(C(C(C(=O)OC)C)=O)CC2)CCC2(CC1)CC(OC)C2 N1(C(C2CCN(C(CN(C)CC)=O)CC2)=O)C2CCC(NC(C)=O)C1CC2 C(C(F)C(=O)NCC1CC(O)C1)C1CN(C(C(C)=C2CC2)=O)C1 c1(C(=O)NCCCCCCNC(C2(CC)CCNC2=O)=O)ccc2nsnc2c1 N1(C(C=Cc2c(C)n(C)nc2)=O)CCCC2CCN(C(C3CCSCC3)=O)CC12 N1(c2ncnc3scc(C)c32)CCCC(C2CC2NC(c2ccnc(O)c2)=O)C1 C1(C(=O)NCCC(C)(C)F)C(C2CC2)CCN1C(=O)C(F)C1CCCC1 C12(NC)CCCC1CN(c1nc(-c3ccc(OC(C)=O)cc3)no1)C2 c1(OC)ncnc(C(N2CCN(C)CC2CNC(=O)CN2CC=CC2)=O)c1F O=C1CCC(C(=O)NC2CC2C(=O)NNS(N)(=O)=O)C1 c1(C(=O)OCC(C)OC)ccc(C2C3CC2O3)cc1.C(=O)N(C)C1CC1.OC c1(CNC(C=C(C)C(F)F)=O)ccc(CN(C)C(c2cncnc2O)=O)cc1 C1(N(C(=O)C(F)CC2CC2)C)CCCN(C(c2c[nH]nc2F)=O)C1 c1(OC)ccc(C(N2CC(CNC(=O)CC(C)C(C)C)C(O)C2)=O)cc1N N1(C(C2N=C(C)SC2)=O)CCCC(N(C)C(C2CC3(C2)CC3F)=O)C1 c1(CCC)nc(C(=O)N(CCCNC(C2CCS2(=O)=O)=O)CC2CCCC2)cs1 N1(C(C=Cc2c(C#N)cccc2)=O)CCN(C(=O)Cc2cc[nH]n2)C2COCC12 C1(C(C2CCCO2)C)CCCN1C(C1CCN1C(=O)OC(C)(C)C)=O C12(C(=O)NCCCOCCOC)CC1CN(C(=O)C(F)C1CCCC1)C2 c1(C(=O)NCC)csc2c1CCN(C(=O)CN(C1CC1)CC)C2 c1(NC(C2C(CNC)C2)=O)ccc(C(N2CCCC2C(C)(C)C)=O)cc1 C(CCCCCC(=O)OC)(c1n(C(CNc2ccc(F)c(Br)c2)C)nnn1)OC C1(NC(C2CN(C(N)=O)C2)=O)Cc2ccccc2N(C(=O)CCC2(O)CCC2)C1 C1(C(=O)N(CC(c2ccccc2)O)C2CC2)CCN(C(c2cnco2)=O)CC1O c1(CC2C(C(=O)NCCn3cc(CC(=O)OC)nn3)C2)ccc(SC)c(F)c1 Cc1cc(C(=O)NCCCOc2ccc([N+](=O)[O-])cc2)c(N)c(C)c1 C1(NC(C2CC(C)(CC)C2)=O)COC2(CCN(C(=O)Cc3cnns3)CC2)C1 CC1CC(NC(c2cnc[nH]2)=O)CCN1C(c1cn(C)nc1Br)=O N1(CC(=O)NC2CC(C(C)(C)COC)C2)CCC2CC(c3ccc(F)cc3)C2C1 c1(C(N(C2CCCC2)CCNC(CCC#C)=O)=O)cc(C)nc2ccc(Cl)cc12 C1(CC)C(NC(c2ccc(=N)[nH]n2)=O)CCCN1C(=O)CC1CCCC1O c1(Cn2cc(CN3CCC(C(=O)NC)C3)nn2)ccc(Cl)cc1 Cc1nc(C(N2CC(CCCCNC(C3(CO)CC3(F)F)=O)C2)=O)c(C)o1 C(=O)(CCS(=O)(=O)C1CCCC1)NC(C)CN(C(=O)CSC1CCS(=O)(=O)C1)C C#CCC(C)(C)CNC(C1(CC)CN(C(=O)CCCCC)C1)=O CC1CN(C(C2CC(=O)N(C(C)(C)C)C2)=O)CCC1CNC(=O)CC1CC1(Cl)Cl C1(=CC(=O)NCC2(O)CC(C(=O)NCC3COC(=O)C3)C2)CCCCC1 C1(NCNC(=NCC)NCc2cc(CC)on2)CCC2COCCC2C1 N1(C(C(C)C(C)(F)F)=O)CCN(C(c2ncn(C)n2)=O)C2CCCC12 CC(C)C(CNC(c1n[nH]c(O)n1)=O)NC(C1(F)CCCC1)=O N1(CC(N2CC3CC3(C(=O)NCc3ccnc(O)c3)C2)=O)CCS(=O)CC1 C1(NC(C2CCN(C(C)=O)CC2)=O)CC2CCC(C1)N2C(c1ccccn1)=O C(=O)(C(F)CC(C)(C)C)NC(CC(C)C)CNC(=O)C(CCO)N(C)C C(=O)(CCCC(=O)NOC(C)(C)C)NCC1CC(NC(C=CSC)=O)C1 c1(C(=O)NCC2C3N(C(C=CCC)=O)C(CC3)C2)c(F)ccc(O)c1F Cc1onc(-c2ccncc2)c1C(=O)NCC1CC(NC(=O)C(F)(F)Cl)C1 c1(NCC2(COC)CC2)nc2ccc(S(=O)(=O)NC3(C)CC3)cc2s1 c1(C(=O)NC(CN(C(=O)CC(C)c2ccco2)CC)C)cncc2nc(C)[nH]c12 c1(-n2ncc(C(=O)NCC(O)CNC(C3CC3C(F)F)=O)c2)ccccc1F C(=O)(CC(C)(O)C(F)(F)F)N1CCC(NC(C(COCC)(C)C)=O)C(O)C1 N1(C(C2C(c3c(C)cc(F)cc3)C2)=O)CC2CCC1CN2C(=O)C1=CCCOC1 Cc1nc(NCc2csc(C)c2C)cc(=NCC2CC3CCCC3C2)[nH]1 C(CS(=O)(=O)CC(=O)NCC1CCC1NC(C1CCC(=C(F)F)CC1)=O)OC C1(C(N2C(C)CN(C(=O)CO)C(C)C2)=O)CC12C1CC3CC(C1)CC2C3 c1(C(N2CC(NC(C(CC)C(=O)OC)=O)CC2(C)C)=O)ccc2c(c1)OCC2 C1(NC(c2n(COC)ncc2)=O)CC(NC(=O)CN2CCC(C)C2)CC1O c1(CC)ccc(Br)cc1C(=O)NC(c1cn(-c2ccc(Cl)nc2)nn1)C Cc1cc([N+](=O)[O-])cc(Br)c1C(=O)N(C1CCNC1=O)C CC1CCc2[nH]nc(C(=O)NCC34CCCC3CN(C(=O)CSC3CC3)C4)c2C1 C1(NC(c2cc(=O)cc[nH]2)=O)CN(c2nc(Cl)ncc2Br)CC2(CCC2)C1 CCC(CC)C(C)C(=O)Nc1cnc(C(C)C)nc1C(F)(F)F C1(CC)(CC)CC(NC(=O)C(C)(CO)SC)CN1C(c1cnc(OCC)s1)=O CC1Cc2ccc(F)c(Br)c2CN1C(C1CN(C)CC1c1ccccc1)=O CC1=C(C(=O)N2CCC(CO)C(NC(=O)C(C)CN(C)C)CC2)C(C)(C)CCC1 C(CC(C)C)(C(=O)N1CC2(CC(NC(=O)CC3CCCN(C)C3)C2)C1)NC(C)=O N1(C(C=CCCC)=O)CCC2(CCCN(C(c3cc(OCC)ncn3)=O)C2)CC1 c1(C(CC)=O)ccccc1C(=O)NCCN(C(=O)C(c1c(C)noc1C)C)C N1(C(=O)CCC2CC2(Cl)Cl)CC2CCN(C(c3ccc4c(c3)OCO4)=O)C2C1 C1(C)(CC(=O)N(C(CNC(Cn2ncc(CC)c2)=O)C2CC2)C)CCCCC1 CC1(C)Cc2c(C(=O)NCCCNC(C3CC(F)C3)=O)cccc2O1 C1(C(N(C2CN(C(c3cc(Cl)n[nH]3)=O)CCC2O)C)=O)CCCCNC1=O c1(OC)cc(CC(=O)NC2CCC(NCc3ccnc(F)c3Cl)CC2)ccc1O c1(C2(C(N(CC(C)(C)CNC(c3sccc3F)=O)C)=O)CC2)ncccc1F C(=O)(CCCS(=O)(=O)N1CCCC1)NCC1N(C(C(CC)O)=O)CCC(C)C1 N1(C(COCC#C)=O)CC(=O)NC2CN(C(=O)CC3CC3COC)CCC12 CC(CCC(C)(C)C)C(=O)NC(CC(=O)N1CC(C)(F)C1)C(F)(F)F C1(C(N(C2CCCC2)CCNC(c2cc[n+]([O-])cc2)=O)=O)C(F)(F)C12CC2 C1(NC(C(C2CCOCC2)C)=O)CCCCN(C(=O)CC2CCOC(C)(C)C2)C1 Cc1cccc(F)c1CC(=O)NCC(F)CNC(=O)C=CC(C)C C1(CNC(C(C)CCO)=O)CN(C(c2cn3ccccc3n2)=O)CCC1(C)C C(=O)(NN1CCCC1C(=O)N(C)OCC(F)(F)F)C1(CC)CNC(=O)C1 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1(C)CCC(NC(C=CCCC)=O)CC1 c1(C(=O)NC)cccc(CN(C)CCNC(=O)C(c2ccc(Br)nc2)(C)C)n1 Cc1noc(Cl)c1CCC(=O)NCC1(NC(=O)CCCCO)CCCCC1 C1(C)(C(=O)OC)CC(N=c2ccn3nc(C(F)(F)C(F)(F)F)nc3s2)C1C(=O)OC C1(NC(c2cnco2)=O)(CF)CCN(C(c2c[nH]cc2C(F)(F)F)=O)C1 n1(CCC)nc(-c2ccc(Cl)s2)nc1CC1CCC2CC12 N(C(=NCc1ccco1)NCC1CCCC12CC2)Cc1nnc(C)s1 Cn1c(C(c2ccccc2)NC(=O)NCC(c2ccc(O)cc2)O)cccc1=O CCC(CC)(CCNC(=O)C(C)OCCOC)NC(=O)Cn1ccc(=O)cc1C C1(C(=O)NCc2cccc(OC)n2)C2CCC(C2)N1Cc1ccc(SC)nc1 c1(C(=O)NCC(=O)NCCCCN(C(=O)C(F)n2ccnc2)C)ccccc1 Cc1nc(CNC(c2ccc(O)nn2)=O)oc1C(=O)NCc1nc(C#N)cs1 C1(CNC(C(C)Sc2ccc(OC)cc2)=O)CCCCCN1C(=O)CSC1CC1 C1(c2n(CCSCC)nnn2)(NC2CCC(C(=O)OC)CC2)COC2(CCCC2)C1 CCCCCCC(=O)N(CCC(C(C)(C)C)NC(C1CN2CCN1CC2)=O)C CCC(CCC(=O)NC(C)CCCC(C)C)NC(=O)CC=Cc1ccccc1 C=CC(C)(CC)C(=O)N1CCN(C(=O)CNC=O)C(c2ccncc2)C1 CC(C)CCC(=O)C(=O)NC1CCCCC1CNC(=O)Cc1nccs1 c1(C(N(C2CCN(C(=O)CCc3cnn(C)c3)CC2)C)=O)nc2ccccc2o1 c1(N(C)C)ccc(C(=O)NC2CCC2CNC(c2ncoc2C(F)F)=O)cn1 N1(C(CN(C(=O)CCCc2cccs2)C(C)(C)C)=O)CCC(O)(CC2CC2)C1 c1(OC)cccc(C)c1CN1CC(C(O)C(=O)O)C1 n1(C(C)C(=O)OCCCC2CC2)cc2ccccc2n1 c1(CC)ncc(C(N2CC(CNC(C3CC3CC(C)C)=O)C(C)C2)=O)c(C)n1 N1(C(CCC=CC(C)C)=O)CCOC(CCNC(=O)COC2CC2)C1 CCCCCCC(C)COC(C)=O.C12CN(CCO1)S(=O)(=O)C2 CCC(C)(O)C(=O)NCC1CCN(C(c2cncc(C(=O)OC)n2)=O)C1 CC(C)(C)CCCC(=O)NC1CC(NC(=O)C(c2ccccc2)C2CC=CCC2)C1 c1(C(C)C(=O)NC2(CCNC(c3nsnc3O)=O)CC2)cccc(F)c1 N1(C(CC(CC)(C)C)=O)CCCC2(CCCN2C(=O)C#CC2CCOC2)C1 N1(C(CN(C2CC2)CC)=O)CC(C(N2CC[Si](C)(C)C2)=O)C(C)C1 c1(NCC(C)CNC(c2cc(S(N)(=O)=O)c[nH]2)=O)nc(Cl)nc2c1ncn2C N1(C(CSc2c(C)n[nH]c2C)=O)CCOCC(NC(C2(C)CC2(F)Cl)=O)C1 c1(C(N2C(CNC(c3ccn(C)n3)=O)C=CC2)=O)cc([N+](=O)[O-])c(Cl)cc1Cl C1(C(=O)NCC(CNC(C(C)(C)C(N)=O)=O)O)CC2COCC(C1)C2 CC1CC(NC(c2cnn(C)n2)=O)CN1C(=O)C(c1cccc(F)n1)(F)F c1(NC(CONC(=O)OCc2ccc(Cl)cc2)=O)onc2ccccc12 O=C(CCC(F)F)NC1(CCNC(c2cc(C3CCC3)on2)=O)CC1 CC1=CCC(C(C)CC(N2CCCC(C(C)NC(=O)C(C)C3CCC3)C2)=O)CC1 C1(NC(=O)CNC(C2CCC2)=O)CCN(C(c2cnns2)=O)CC1O C(=O)(C(F)(F)CCn1cc(CCc2ccsc2)nn1)NCc1nc(SCC)sc1 c1(C(=O)OCC)coc(C(=O)NCCN(C(C2CCC(CC)C2)=O)C)n1.C1(S)CC1 N1(C(CCC(=O)OC)=O)CCCOC(CNC(=O)C(C)(C)N2CCCC2)C1 Cc1ccc(C#N)c(N2CCCC(CNC(C3CCCCC3)=O)C2)n1 Cc1ccc(F)cc1C(N1CCN(C)CC1CNC(=O)C(CO)C(C)C)=O N1(C(Cc2nc(C)c(C)s2)=O)C2CCCC1CC(NC(C1(C(F)(F)F)CC1)=O)C2 CC1CCc2c(F)cccc2C1NC(=O)CCC1CCCCC1=O C1(CC(=O)NC23CC(NC(c4nc(C(=O)OC)sc4)=O)(C2)C3)CCC(=O)NC1=O CCCC(C(=O)NCCn1cnc(C(N2CCC(O)(C(F)F)C2)=O)c1)OC C1(CN(C(=O)Cn2cc(Cl)cn2)C)CCCN(C(C2CCCC(N(C)C)C2)=O)C1 c1(C(C)(C)C)ccc2c(c1)NC(=O)C2NC(=O)C(N)CC1CC1 c1(C(=O)NC(CC)CNC(=O)CC2CC(F)(F)C2)cccc2ncc(Br)n12 C(=O)(C1=CCCOCC1)NCCC1CC(NC(c2ccn3cncc3c2)=O)C1 C(c1ccc(F)cc1)=CC(=O)NC1C2CN(C(c3cccc(N(C)C)c3)=O)CC21 C1(C(=O)NC(c2ccncc2)CCC)Cc2ccccc2CN1CC(C)O c1(C(N2C(C)CCC(NC(C3(CC)CC=CC3)=O)C2)=O)cc2n(n1)CCNC2=O n1(C(C(=O)NC(CNC(CCC(=O)NC)=O)C(C)C)C)c(C)cc(O)cc1=O C1(C(=O)NCCS(C)(=N)=O)CCOCC1NC(C1CCNC1=O)=O C(=O)(CCCC(C)(C)C#N)N(CC(CC)C(=O)NCCCSC)C N#Cc1cnc(NC(N2CCCC(NCC3CC3(F)F)C2)=O)c(F)c1 C#Cc1c[nH]nc1C(=O)N(c1cc(C(=O)N(CC(C)(C)C)C)n[nH]1)CC(C)C C1(C(N2CCC(N(C(=O)C(F)=C3CCCC3)CC)C2)=O)CC(C)(C)OC1(C)C C1(C#N)(C(=O)NCCn2ncc(C(N(C(C)CCO)C)=O)c2)CC2CC2C1 Cc1ncnc(C)c1C(=O)NC1CCCC1NC(C1(C)C=CCC1)=O c1(C(N2CC=CC(NC(=O)C3=CCOCC3)C2)=O)c(Cl)ccc(Cl)c1O Cc1cnn(C)c1C(=O)NCC(CC1CC1)CO c1(C(=O)NC(CN(C(C(C)C2CCC2)=O)C)C)cc[nH]c1C1CC1 Cc1nc2c(s1)CN(C(=O)CCC1CCCN1Cc1ccc(O)cc1Br)CC2 c1(N2CCC(C#N)(N(C)C)C2)c(-c2ccccc2)[nH]c2c(Cl)cccc12 CN=c1cc(C(N2CCC(C(=O)NCC(O)CC(C)C)(C(C)C)C2)=O)cc[nH]1 c1(C(=O)NCC(CN(C(CCC(C)OC)=O)C)O)cccc2nc(C(F)F)sc12 C1(NC(=O)Nc2c(OCC)cc(C)s2)CCCN(C2CCCCO2)C1=O N12C(CC3CCCCC13)C2=O.N1(C(=O)OC(C)(C)C)CC(O)(CCS(C)(=O)=O)C1 C12(CS(=O)(=O)NCC)CCCNC1CCC2.C12CCCCN1C(=O)CC2 Cc1cc(C)c(C(N2CCCCC2C(C)NC(c2nc(C3CC3)cs2)=O)=O)[nH]1 Cc1cc(Cl)c(C(N2CC(C)(C)CC2CNC(c2nc(C)n(C)n2)=O)=O)cc1C c1(C(=O)NC2CC(NC(=O)C(F)C3CCOC3)C2)ccc(C2CCC2)nc1 c1(CN(C(=O)CCN(C)CCOCCO)CCNC(C2(C)C(C)C2)=O)ccccc1 c1(C(=O)NC(CNC(C(CCC)C(C)C)=O)CC)ccc(O)cc1[N+](=O)[O-] Cc1cc(=NCC(C)(C(C)C)NC(c2ccc(F)c(C)c2)=O)[nH]c(Cl)n1 Cc1nc2cncc(C(N3CCC(CO)C(NC(c4cnn[nH]4)=O)C3)=O)c2[nH]1 C1(C(=O)NC2CN(C(C(CC=C)C)=O)C2)CC12CCc1ccccc12 c1(C(N2C(CN(C(c3c(C)coc3C)=O)C)COCC2)=O)cccc(Cl)c1Cl N1(C(CSCC)=O)CCC(C(C)C(=O)NC(c2nc(C)cs2)(C)C)CC1 C(=O)(CC(C)(O)C1CCCCC1)NC(CNC(c1cn(CCOC)nc1)=O)C N1(C(CC2CC(C(=O)OC)C2)=O)CCCCC1CCCNC(=O)CC1CCOC1C C1(C(=O)NC(CNC(=O)COCc2ccncc2)C2CCC2)CCCOCC1 c1(C(N2C(C(N(CCC(F)(F)F)CC)=O)C(C)CC2)=O)cnc(C)[nH]c1=N CCCC(CC(C)C)C(=O)NCC1CCN(C(c2c(C)cnnc2O)=O)C1 c1(OC)cncc(C=CC(N2CCC(O)(C(C)CNC(=O)C3=CCCC3)C2)=O)c1 c1(C(=O)NCCN(C(C2C(OCC)CCC2)=O)C)cccnc1SC(C)C Cc1cc(C)c(S(N)(=O)=O)cc1C(N1CCCCC1CN(C)Cc1cnn[nH]1)=O N1(C(C2(C#N)CCC2)=O)CCC(F)(F)C(CNC(=O)C=C2CCCC2)C1 C1(c2cnc(OC)c(C)c2)CCC2(CN(Cc3cc(F)cc(F)c3F)C2)O1 c1(C(=O)NC2CCC(NC(C(C)OCCOC)=O)CC2)ccc2c(n1)CCCC2 C1(O)(CC)CCCN(C(=O)C(CC2CCC2)NC(c2cc(F)ccc2F)=O)C1 C1(C)(C(N2CC3C(CNC(c4cc(C)cc(F)c4)=O)C3C2)=O)CCCCC1(F)F c1(C(=O)NC(C)CC2(OC)CCN(C(=O)C(C)CC(C)C)C2)cc(OC)nc(Cl)c1 CC1CN(C(c2ncc(F)cc2F)=O)CCC1N(C(=O)C(=O)N(C)C)C C#CCC(CC(F)F)C(=O)NCc1ccc(CCNC(C2(COC)CC2)=O)cc1 C12(C(N3CCC(CNC(C4COC(=O)O4)=O)C3)=O)CC1COC21CCC1 c1(C(N2CCC(N3CCCC(C(C)=O)CC3)C2C)=O)c2c(nn1C)CCCC2 Cc1cc(CC(N2CCC(NC(C3CCCS3)=O)C2)=O)nn1C C1(CNC(C(CC)N(C)C(c2c[nH]c(=NC)o2)=O)=O)CC(=O)N(C)C1 C(=O)(C1SCCc2sccc21)N1CC(OCCNC(C2(O)CC(C)(C)C2)=O)C1 c1(NC(C(N2CCCC2(C)c2ncc[nH]2)c2cc(C)on2)=O)cccc(Cl)c1C c1(C(=O)NCC(COC)NC(=O)CCc2cncnc2)cccc(OC)n1 Cc1ccc(C(=O)NCC(O)CN(C)C(c2cnccn2)=O)c2ccccc12 S(=O)(=O)(c1cc(Cl)ccc1OC)NC(C1(NCC)CCCC1)=O C(=O)(CCCC(=O)NC1CC1NC(=O)C=CBr)Nc1c(C)cccc1 N1(C(C2N(C)CSC2)=O)CCC2(CC1)CCN(C(=O)C(C)(C)C(F)F)C2 Cc1cc(CC(=O)NCC2COCCN2C(=O)Cn2cncn2)cc(C)c1 N1(C(C(C)N(C(c2c(CCC)n[nH]c2)=O)C2CC2)=O)C(CO)CC2CCCC12 C(=O)(C1CCCc2nncn21)NCC1C2CN(C(C(C#C)(C)C)=O)CC21 C1(CNC(C(C)N(C)C)=O)CC(NC(=O)CC(=O)NCC(F)(F)F)CCO1 C(=O)(CCCCCCNC(=O)CN1CCCCCC1)N(C)Cc1csc(=N)[nH]1 c1(C(=O)NC2C(CNC(C3CCCC(OC)C3)=O)C2)cnc2ncnn2c1C N1(C(c2ccc(C3CC3)cc2F)=O)C2CCC1CN(C(C13C=CC(CC1)C3)=O)C2 CN1CC(C(=O)NCCOCC(=O)NCC2(CO)CCN(C)C2)NC1=O c1(-n2c(C)nnn2)ccc(C(=O)NCC2C3CN(C(C4CC(F)C4)=O)CC23)cc1 Cc1cc(CC(=O)NCC2CN(C(=O)CCn3cccn3)CCO2)cc(F)c1 c1(C(=O)OC)cc(=NC(C)c2cc(F)cc(Cl)c2)[nH]c(Cl)n1 C(C(CNC(=O)CCSCC(C)C)C(F)(F)F)NC(c1nc(C#C)sc1)=O C12CCC1NC(=O)CN(C1CCCC1)C2=O.C(C(CO)C1CC1)SCCO C=Cn1nccc1C(=O)NC(CC1CC1)C(=O)NCCS(N)(=O)=O C1(NC(c2ccn(CCOC)n2)=O)CN(C(=O)C(C)(C)CC#N)CCC12CCC2 C=C[Si](C)(C)CNC1CCN(c2ccc(C(=O)O)cc2)C1 Cc1cc(CC(=O)NCC2(C(C)NC(=O)C(C3CCOCC3)O)CC2)no1 NC1CCCCC1n1cc(C(=O)N(C2CCOCC2)CCCO)nn1 C1(C(N2C(CNC(c3cnc(O)s3)=O)CCCCC2)=O)CCn2c(O)nnc2C1 C1(NC(C2CC(OC)C2)=O)CN(C(c2ccccc2COC(C)C)=O)CC12CC2 N1(C(CSCCNC(C(C)n2ccnc2)=O)=O)CCC(C(C)(C)O)C1 N1(C(C2(F)C(C)C2)=O)CCCC2(CCN(C(=O)C(F)CC3CCOC3)CC2)C1 N1(C(CSC(C)C)=O)CC2(C=C(C(=O)NOCCF)CO2)C1 C(=O)(C(C)(C)C(C)CC)NCc1cncc(C(=O)NCCC(=O)OCC)c1 c1(C(=O)NC2CC(C)(NC(C(CCCC)CC)=O)C2)cnn2cccc(C)c12 c1(CNc2ncnc(N3CCCC(SC)C3)c2C)cnn2ccncc12 c1(C(N2CC(CNC(C(C(C)O)(F)F)=O)N(C)CC2)=O)cccn2ncnc12 CC1(C)C=C(C(=O)N2CC(CCNC(c3cc4sccc4s3)=O)C2)C1 c1(C(N2CC3C(NC(C(C)n4ccnc4)=O)(C3)C2)=O)cc2ccncc2s1 c1(CCNC(Cn2c(COC)nnc2-c2ccc(Cl)cc2)=O)ccccc1O C1(OC)CN(C(=O)COC(F)(F)F)C(C)(CNC(c2ccoc2C(F)(F)F)=O)C1 NS(=O)(=O)c1cc(C(=O)OCC2CC(F)(F)C2)ccn1 c1(-n2cc(C(C)(C)NC(CCN(C(C)=O)C(C)C)=O)nn2)ccc(F)cc1F Cc1cc(F)c(N)cc1C(N1CCC(CNC(=O)C(C)C2CCCC2)C(C)C1)=O c1(C(CC(=O)OC)NC(=O)C(=O)NC2CCN(C)C(C)C2)ccccc1[N+](=O)[O-] c1(SC)cnn(C)c1C(=O)NCC(CC(C)C)NC(c1ccncc1Br)=O c1(-c2cn(C)nc2)nn(C)cc1NC(C1CC12CN(C(=O)COCCCF)C2)=O C1(NC(C(CC(C)C)n2ccnc2)=O)CN(C(C2CC2C(F)F)=O)CC12CCC2 c1(C(=O)NCC(CNC(c2c(COC)scc2)=O)O)ccccc1-c1ncc[nH]1 c1(CC(N2C(C(C)(C)NC(c3scc(C)c3)=O)CCC2)=O)ccc2nonc2c1 C1(CCNC(c2ccnc(F)c2)=O)CSCCN1C(c1ccncn1)=O C1(C(=O)NCC(C(C)C)NC(C=CC=CCC)=O)CCn2ccnc2C1 Cn1cc(CNC(CNC(c2scnc2Cl)=O)C2CCC2)c2cccnc12 Cc1cc(C)c(CNC(=O)NC2CC2Cc2ccccc2)c(O)n1 c1(C(N2CCC(NC(C3ON=C(C)C3)=O)C2C)=O)ccc2occ(C)c2c1 O=C(C1=CCCOCC1)NCC1(CNC(c2ncccn2)=O)CCCCC1 c1(C(=O)NCC2CCC2c2cccs2)cc2cccc(Cl)c2cn1 c1(C(N2CC(CNC(C(C)CC(C)(F)F)=O)C(C)C2)=O)ccc2c(c1)CNC2=O C(=O)(C1=CCC(C)(C)CC1)N1CC2OCC(NC(CCc3onc(C)n3)=O)C2C1 C1(C(N2CCN(C(CCC(C)(C)O)=O)C(CCO)C2)=O)CC2CCCC(C1)C2=O Cc1cc(CN2CC(C3(NC(C4CC(=O)N(C)C4)=O)CC3)C2)cc(C)c1 N1(CC)CC(CNC(C2CCCCC2CNC(=O)C(C)(C)CC2CC2)=O)OC1=O C(=O)(C1CCCCc2ccccc21)N(C)CC1(NC(c2sccc2C#N)=O)CC1 N1(C(C(C)CC(N)=O)=O)CCCCC2(CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 C12(NC(c3cc(C)ncc3)=O)CCCC1N(CC(C)CC(C)C)CC2 C1(Nc2nnc(CC(N3CCCC(O)(C(C)C)C3)=O)o2)CCc2nnnn2CC1 C1(NC(CC2(CSC)CC2)=O)CN(C(c2cc(C(F)F)no2)=O)CCC1C(F)(F)F C1(C(=O)NCC2CN(C(c3ccc(CCC)cc3)=O)CC2C)CCN(C)C(C)C1 CCCC(C)CC(=O)NCC1(NC(=O)C(C2CCC(=O)N2)C)CC1 C(CCC1CC1)(C(=O)N(C1CSC1)C1CC1)NC(=O)CC1COCC1O C(=O)(N1CCC(C(=O)NC(C)C(C)C)O1)c1cccc(OC)n1 C(C1=NOC2CCCC12)NC(C(=O)NCC(Cc1ccc(C)s1)OC)=O C1(NC(C(=O)NCC2CCCCC(=O)N2)=O)CC2CSCC(C1)C2 N1(C(CN(C(=O)Cc2ncn(C)c2C)CCOC)=O)CC2CCCC1C2 C1(NC(c2nnn(C)c2N)=O)CCN(C(=O)Cc2cccc(C#N)c2)CC1(C)C C(CC(C(C)(C)C)NC(c1csc(C(N)=O)n1)=O)N(C)C(c1[nH]cnc1C#N)=O CCCCC(C(=O)NCCc1ccc(F)nc1)NC(=O)C(C(C)(C)C)OC C(C(C(=O)NCCC1CCCO1)C(C)C)NC(c1c(C)cccn1)=O C1(O)(C(CC)C)CCN(C(C2(CNC(c3cc(CC4CC(C)C4)on3)=O)CC2)=O)C1 CC1(C)CN(C(=O)CC2CCC3CC3C2)CC1NC(c1cccc(F)c1N)=O C(=O)(CCCC(=O)OC)N1CCC(C)(C(=O)NC(CCC)c2ccco2)C1 C1(C)(C(=O)NCC2CN(C(CN(C(C)=O)C)=O)CC2(C)C)CCCCNC1=O Cc1cccc2[nH]cc(CC(=O)NC3CC3CNC(=O)Cc3cn(C)nn3)c12 N1(C(c2ccc(OC)nc2C)=O)CCN(C(=O)CCC2CC2(F)F)C2(CCC2)C1 CC1CN(C(=O)Cc2cnoc2)C(C)CN1C(=O)CN1CCCC1C c1(C(N2CCC(N(C(=O)CCC3CCCO3)C)C2)=O)ccc2nc(O)[nH]c2c1F C1(C(=O)Nc2ccc(Br)cc2F)CN(C(c2cncnc2)=O)CC(F)(F)C1 CC(CN=c1[nH]c(C(F)F)nc(=N)[nH]1)N(C(=O)C(F)(F)c1nccs1)C C1(C(=O)NC)CCCC1N=c1[nH]c(=NCc2cccc(COC)n2)[nH]c2ccsc12 C1(C(N(CC(COC)(F)F)C)=O)C2CCC(C2)N1C(C1CC1OC)=O N1(C(C2(C=C)CCC2)=O)CC(NC(=O)CC2CCOC2)C(C)(C)C1 c1(NCCC(=O)OCC)ncccc1C(=O)CN(c1ccccc1)C C1(C(=O)NCC2CCN2C(=O)C=CC2CCC2)CCCN(c2ccccn2)C1 C=CCCCCCCCC(=O)N1CC(C(=O)C(C)C(O)CC)(O)C1 C1(CNC(Cc2c(C)cc(F)cc2)=O)COC(C)(C)CN1C(C1CC(CF)C1)=O c12ccc(nc1)C(=O)NCCN(C(c1ccc(CC)[nH]1)=O)CCO2.C#CCOC c1(C(N2CCC(C(C)NC(=O)Cn3ncnn3)C2)=O)ccc(Br)cc1O c1(C(N2CC3C(C(=O)Nc4cnc(OC)o4)C3C2)=O)ccc2nc(C3CC3)[nH]c2c1 c1(C(N2CCC(N(C(c3nccs3)=O)CC)C2)=O)cnc2c(F)cccn12 C1(C(=O)NCCCN(C)C(c2cccc(C(C)(C)C)n2)=O)OC2CCC1C2 C1(OC)(CNC(c2cc(C(N)=O)cs2)=O)CCN(C(c2ncc(C)cc2F)=O)CC1 c1(NC(C)=O)cc(C(=O)NC2CC(NC(c3cc(Br)cnc3Cl)=O)C2)ccc1C C1(NC(c2ccc(Cl)o2)=O)CCC2CCN(C(=O)C3=CCS(=O)(=O)C3)C12 Cc1ccc(NC2CCCCC2CN)cc1-n1cnnn1 c1(COC(C2CCCC(F)C2)=O)c(O)cccc1Cl C(C(C)(C)C)N(C)C(C1CC(NC(=O)COC2CC2(F)F)C1)=O c1(C(N2CC3N(C(c4c(CC)occ4)=O)C(CC3)C2)=O)cc(S(C)(=O)=O)oc1C c1(OC)ccc(C)cc1C=CC(=O)NC1CC2CN(C(c3ccsc3)=O)CC2C1 CCC(C)CC(N)C(=O)N(C(C)(C)C)Cc1c(C)cccc1C c1(OC)ccc2c(C(=O)NC3CC3(C)C(F)F)n[nH]c2c1F C(c1cc(Cl)ccc1Cl)=CC(=O)N(C)CC1C2CN(C(c3nc(C)[nH]n3)=O)CC21 CC1(C)CC(O)CN(C(=O)CC2(NC(=O)CN3CCCCC3=O)CCC2)C1 c12cccc(c1)CO2.C1(NC(C(=O)NCCC(=O)OC)=O)CCCC(C)OC=C1 Cc1nn(CC(=O)NC(C)(CNC(=O)CC(O)CN(C)C)CO)c(C)c1[N+](=O)[O-] C1(N(C)C(c2cn(C)cn2)=O)CC2CCC(C1)N2C(c1ccc(C#N)o1)=O c1(NCC(C)(C(C)C)NC(c2c(C)noc2)=O)cc(Cl)ccc1[N+](=O)[O-] c1(CC(=O)NC(C(C)C)CNC(c2csc(Cl)n2)=O)ccc(-n2cnnn2)cc1 CC(C)CC(C)(CNC(C1(C)CCCS1)=O)NC(C1CN(S(N)(=O)=O)C1)=O c1(C(=O)NCC(C)CN(C)C(C2CC2CF)=O)cc2n(c1)CCS(=O)(=O)C2 C1(CNC(C2C(C)C2)=O)C2CCC(C2)N1C(=O)CCN1CCCCC1=O C#Cc1ccnc(C(=O)NCC(O)C(=O)NCc2cc(C)cc(F)c2)c1 Cc1ccc2cc(C(N3CCC4(CCN(C(=O)CC5CC5)C4)C3)=O)ccc2n1 c1(C(N2CC(NC(C3C(C)C3)=O)CC23CCC3)=O)ccc(S(C)(=O)=O)cc1N C1(C(N(CCCC#C)CCO)=O)CCCC(NC(=O)CC2CCC(=O)N2)C1 C(=O)(CCCc1cccs1)NCCC(C1CC1C(=O)NC1(c2cnn[nH]2)CC1)C CC1CS(=O)CCN1C(=O)CNC(=O)CNC(C1CCCC(=O)CC1)=O C1(C(N(C)CCOCCC(=O)NCc2ccnc(O)c2)=O)CC2(CCC2)C1 c1(C(=O)NCC2(O)CC(NC(C3C(C(C)C)C3)=O)C2)ccc(S(N)(=O)=O)o1 C(=O)(CC(C)CC(C)C)N1CC(CC(C)NC(Cc2cc(CC)no2)=O)C1 c1(C(CC)C(=O)NC(C)CCNC(C2CC2F)=O)ccc(OC)cc1 c1(C(N(C(C)CNC(=O)C(C)OCC(F)(F)F)CC)=O)c[nH]c2nccc-2c1C C(CC(C(N)=O)NC(c1cc(CNC(c2cscc2C)=O)nn1C)=O)OC C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(NC(c2cncc(C#C)c2)=O)C1(C)C c1(C(C(C)C)NC(c2ccncc2)C(F)F)cnn(C)c1.C(C)(C)(C)NC(=O)O C(C(=O)N=c1[nH]onc1C1CCC1)c1c(F)ccc(OCC)c1 O=S(=O)(c1c(Cl)cc(Br)cc1Cl)NC1CC12CCN(Cc1c[nH]c(Br)c1)CC2 C12(NC(Cc3cc(C)[nH]n3)=O)CCCC(NC(=O)C=C3CCN(C)CC3)(C1)C2 C#Cc1cccc(C(=O)N(C)CC2CCCCN2C(=O)C=CC(=O)N(C)C)c1F C#Cc1nccnc1NC(c1c[nH]nc1C(=O)NC(C)C(=O)OC(C)(C)C)=O C(CN=c1[nH]ccc(=NC2CCCC(n3ccnc3)C2)[nH]1)=C(C)CC1CC1 C(N=C(NC(C)C=C)N1CCC(Br)=C(C)C1)c1ccc(OCC=C)nc1 C1(F)(CNC(CNC(C(CC)C)=O)=O)CCC(NC(c2cnn(C)c2)=O)C1 C1(CC)CN(C(C2CC2C2CC2)=O)CCN1C(c1cscc1OC)=O N1(C(C)=O)C2CCC1CC(CCN(C(=O)Cc1cc(Cl)cnc1C)C1CC1)C2 Cc1occc(=O)c1OCC(=O)NCC(C)(C)NC(=O)C=C1CCC1 C(=O)(C(F)C(C)CNC(=O)CCCN(C)C(C)C)N1CC(CCC)OCC1 N1(C(Cn2c(C)cnc2)=O)CC(NC(=O)C(O)C2CCC2)CC1C c1(CC)ncc(Cl)c(C(=O)NC2(C)CCN(C(=O)Cc3ccn(CC)n3)C2)n1 N#Cc1ccccc1C=CC(=O)NCCNC(=O)CCC1CCCC(O)C1 C(=O)(CCC(=O)C1CC1)N(CC(C)N(C(C=CC)=O)C)C CC(O)CCC(=O)NCC1(CNC(=O)CC2(O)CCCOC2)CCCC1 c1(C(N2CCOCC(C)(C(=CC(=O)NC)C)C2)=O)cc2c(nc1O)CCCC2O c1(-c2cn(CC(CCNC(CCOC)=O)(F)F)nn2)ccc(Cl)c(F)c1F CC1CC(C(=O)NCC2CC3(CCC3)C2)N(C(=O)CNc2ccccn2)C1 N1(C(c2cn(CCC)nc2)=O)CCCC(F)(CNC(=O)CC2CCCC2O)CC1 C1(CNC(C=COCC)=O)CCC2(CCN(C(c3cc(CC)on3)=O)CC2)CO1 C(CCC(C)CC(=O)NC1C2CC1N(C(c1cncc(C)c1Cl)=O)C2)=C(C)C CCCCC(CNC(c1sc(C)nc1C)=O)NC(C1CCC2CC12)=O Cc1[nH]nc(Cl)c1C(=O)NC1CC(C(C)NC(C2CCCCN2C)=O)C1 CN1CC(NC(=O)C(Cc2ccoc2)NC(=O)C=Cc2cscn2)C(F)(F)C1 CC(C)C#CC(=O)NC1(CCNC(=O)C(C)CC2CCCO2)CCC1 c1(COCCCOCC(=O)Nc2ccccn2)noc(C2CCCO2)n1 N1(C(C=CCCC)=O)CCC(C2(NC(=O)CCC(C)CC)CC2)CC1 N1(C(c2ccc([N+](=O)[O-])s2)C(=O)NCC=C)CCCC1C1CCCCO1 C12(C(=O)NC(CC)(CNC(=O)C=CC(C)(C)C)CC)CCCN1S(=O)(=O)CC2 c1(C(=O)NCC(C)O)c([N+](=O)[O-])cnn1CCN(C)C.c12ccc(cc1)SC2 C(CCC)(C(=O)N1CCCC1C1CCCN(C(c2n[nH]cc2Cl)=O)C1)=CCC C(=O)(C(C(C)C)C(C)C)N1CC(COC)(NC(=O)C(c2ccccn2)C)C1 CC(CN(C)C(c1csc(O)n1)=O)C(=O)N=c1ccn(C)[nH]1 C(=O)(C(C)(C)CCNC(c1cnn2c1OCC2)=O)NCc1c(CC)c[nH]n1 CCC(C)(C)C(=O)C(=O)N1C(C(=O)NCC2CSCCO2)CC2CCCC12 CC1(C)CCC(CCNC(=O)CCOCCNC(C2CN(C(C)C)C2)=O)O1 c1(C(=O)NCC2(OC(C)C(=O)NCc3ccco3)CCC2)c[nH]cc1C1CC1 N1(C(Cn2nnc(C)n2)=O)CCC(C2CC2)C1CNC(=O)CCC(=O)NC1CC1 C(C(C)(CC(C)C)NC(=O)CC1CC(C(=O)OC)C1)NC(C(CC=C)C)=O c1(NC(CS(CC)(=O)=O)C)ccc(S(=O)(=O)NC2CN(C)C3(CCC3)C2)cc1Cl C1(C(N(CCC)CC2CC2)=O)COCCN(C(C2CCCC2C(C)C)=O)C1 c1(C(=O)NC2CCN(C(CCCOC)=O)CC2C)c(F)ccc(C#N)c1F C(=O)(C(COC)(CC)CC)NCC(C(=O)NCC(CCC)OC)(C)CC Cc1nn(C)c(Cl)c1CC(N1CC2(NC(=O)CCc3nc[nH]n3)CC1C2)=O CC1C(NC(C2CC(F)C2)=O)CC2CCC1N2c1nc2ccc(C(F)(F)F)cc2s1 c1(CNC(N(C(C(CC)C)C)CCO)=O)nnc2ccccn12 N1(C(c2c(C)csn2)=O)CC2CCC2(CNC(=O)C(C)CN(C)C)C1 Cc1ncn(O)c1C(=O)NCC(O)CCNC(c1n[nH]c(C(C)(C)C)n1)=O N1(CCNC(=O)CCN(C(=O)CCc2ccccn2)CCO)CC2CCC1C2 CCCCCC(C)CC(=O)NCCCN1CC(C)OC(C)C1 c1(C(N)=O)c[nH]c(C(=O)NCC2CC(O)(CNC(C3CC3F)=O)C2)c1 C(c1cccc(F)c1F)=CC(c1nnc(S)o1)=O N1(C(CC(=C)C)=O)C2CCCC1CC(NC(=O)C1=CCCOC1)C2 Cc1sc(Br)c(C(=O)NCC(C(C)C)NC(c2c[nH]nc2C2CC2)=O)c1C Cc1ccn2ncc(C(=O)NC3(CNC(C4CC5CCCCC5C4)=O)CC3)c2c1 Cc1nnc(CCCC(=O)NCC(F)CNC(C2CC=CCO2)=O)n1C C1(C(=O)NCC(CC)(CC)NC(c2c(OCC)scc2)=O)CC(C(=O)OC)=NO1 C1(N(C(C(C)Nc2ncc(C)s2)=O)C)(C(=O)O)CCN(C)CC1 C1(OC)CCCC(CC(=O)NC2C3CC2N(C(C2CC4(C2)CC4F)=O)C3)C1 N1(C(c2c(C)nc[nH]2)=O)CCCC(C2CN(C(c3sccc3C(C)(C)C)=O)C2)C1 c1(C(=O)NC2(CNC(C34CC(F)(C3)C4)=O)CCC2)c[nH]c(=O)c2ccnn12 C1(CNC(C2CC(C)OC2)=O)CC(N=c2nc(C3CC3)[nH]s2)C1 CC1CCN(C(=O)C=C2CCCC2)CC1CNC(=O)C(O)CC1CC1 C12(C(=O)NCC(C)N(C(C3C(c4nnc(C)o4)C3(C)C)=O)C)CC(C)(C1)OC2C C1(CC)CCN(C(C2CCC2C)=O)C(C(=O)N(C2CCC(=O)N(C)C2)C)C1 Cc1nc(C(=O)NCCC2CCN(C(C3(N(C)C)CC3)=O)C2)co1 N1(C(C2(O)CCCC2)=O)CCOCC(NC(C2(F)CCOC2)=O)C1 C1(C(N(CCN(C(CCCc2c(C)nc(C)s2)=O)C)C)=O)COCC(C)(C)O1 C(=O)(C(=O)N=c1ncn(C(C)C)[nH]1)NC1(N(C)Cc2ccc(C)cc2)CCCC1 c1(OC)c(C(=O)NC(CNC(c2ccccc2O)=O)C2CC2)nc(O)nc1O c1(C(=O)NCCC2CCN(C(C3(CO)CCCO3)=O)C2)ccnc2nccnc12 c1(OC(C)C)cccc(C(O)C(N2CCOCC2CSc2ccc(Cl)cc2)=O)c1 C(CC(CC)C(=O)N1CCCC1CNC(=O)C(C)(C)c1ccno1)=CC N1(C(c2ccc(Br)cc2F)C(=O)NC(C(=O)OC)C)C2CCC1CN(C)CC2 c1(C(=O)NCC(C2CCCC2)O)cccc2ccncc12.C12CC1NC2=O CC(C)CCCCC(=O)NCc1c[nH]nc1C(=O)NC1CCCCCC1CO CC1(C)CN(C(=O)C=Cc2ccccn2)CC1CNC(C1(C)CCC1)=O C(=O)(C(C)S(=O)(=O)C(C)C)N(CCNC(c1cnn2c1OCCC2)=O)CC C1(C(=O)NC(CC)C(=O)NC)CC(NC(=O)CC23CCCC2C3)C(O)C1 Cc1cc(=NCc2cc(Br)no2)[nH]nc1C(F)(F)F C1(N(C(=O)CCCC2CC2)C)CN(C(=O)C(O)Cc2cnn(C)c2)CC1(C)C C=CC1(C(=O)N(C)CC2(C)CCCO2)CCN(C(c2cccc(C)c2C)=O)CC1 N1(C(CC2(C)CCCC2)=O)CCC(C2CC2)(CNC(=O)CCC(F)(F)F)C1 N1(C(C(CCC)OC)=O)CCC2(CCc3ccccc3C2=O)CC1 C1(C(=O)NC2(CNC(c3c(C(C)C)ocn3)=O)CCOC2)CCC12CCC2 C=CC(C)(C)CC(=O)N1CCSCC1C(=O)NCC1COCCN1C C1(C)(C(=O)NCC(CNC(C(CC=CC)C)=O)(C)C)CCCC(F)(F)C1 C(C(COC)NC(=O)C(F)C1CC(NC(=O)C(O)C2CCCC2)C1)OC CC1(C)OCc2cc(C(=O)NCCCNC(=O)C3=COCC3)ccc2O1 C1(C(=O)NCC2(CNC(=O)CC3CC3)CCC2)(OCCO)CCCCC1 C(C(C)(CC(C)C)NC(c1cnc(S)[nH]1)=O)NC(c1ccc(COC)cc1)=O C1(NC(c2ocnc2C2CC2)=O)CCCN(Cc2cn(C3CCC3O)nn2)C1 c1(C(=O)NC2CCCC(NC(C=CC(=O)N(C)C)=O)C2)ccc(=O)n2c1CCC2 c1(CNC(CCNC(C)=O)=O)ccc2c(c1)CCN(c1nnnn1C)C2 c1(C(N2CCC3C(C(N(C)CC4CCC(=O)N4)=O)C3C2)=O)cnn2c1OCC2 CC1NC(=O)CCC1CNC(=O)C(Cc1cn[nH]c1)NC(=O)CC1CC(=O)C1 N1(C(CN2CCP(C)(=O)CC2)=O)CCCC12CCCN(C(=O)C=C1CCC1)C2 C1(O)(CN(C(=O)C=Cc2cocn2)C)CCN(C(=O)CSCC2CCCO2)CC1 CCC(F)(C(=O)OC)C(=O)NC(C)CC(C)NC(=O)CC1(O)CCC1 CC1CCCCC1(CNC(=O)C1=CCOC1)NC(c1coc(C(F)F)n1)=O c1(SCCC(=O)NCCCN(C(C2C(C)C2)=O)C2CC2)nnnn1C1CC1 Cc1cc(C(N2CC3(CNC(c4ccon4)=O)CCC2C3)=O)c(N)c(Cl)n1 c1(CC)ccc(C(=O)N(C2CCCS(=O)(=O)C2)C)c2c1CCCC2 O=C(N=c1[nH]oc2ccncc12)c1ccc(NC(c2cccc(F)c2F)=O)nc1 c1(C(C(=O)N(CC(CC)(C)OC)C)COC(C)C)cccc(F)c1 C(CCC(C)C(=O)NCC(C)(C)CNC(=O)CNC(=O)CC1CCCC1)OC C(CCC(C)C(=O)NCC1CCC1C(=O)NC(C)(COC)CO)OC N1(C(c2c(C)cccc2)=O)CCOCC(C)(CNC(c2csc(O)n2)=O)C1 C1(NC(C2CCC(F)(F)CC2)=O)C2CCN(C(=O)C=CCn3cncn3)CCC12 Cc1nc(Br)sc1NC(C1C2CN(C(=O)C=CC(=O)NC(C)(C)C)CC12)=O c1(OC)cc(C(=O)NC2CN(C(=O)C(C)CN(C)C)C(C)(C)C2)cc2c1OCO2 C1(NC(c2c(C)nns2)=O)CCC2CN(c3ncc(F)cn3)CC2C1 N1(C(C2(NC(=O)C(O)C3CCC3)C(C)(C)C2)=O)CCC2(CNC(=O)N2)C1 Cc1nc(C2CC2)[nH]c1C(=O)NCCC1CN(C(c2cnc(O)o2)=O)C1 CON(C)S(=O)(=O)c1ccc(C(=O)OCC(C2(C)CCC2)=O)cc1 C1(CCNC(C2(CNC(=O)CCSC)CC(=C)C2)=O)COCC(C)O1 C1(CNC(c2c(C)cc[nH]2)=O)CN(C(C2CCCCN2C)=O)CC1(C)C C1(C(=O)NC(CCOC)CNC(c2cncc(N3CCCC3)n2)=O)NC(=O)OC1C C1(CNC(c2ncn(C)c2)=O)COCCN1C(C1CC(F)(CF)C1)=O CC(C)(CN=c1ccc2ncc[nH]c-2n1)NC(c1ccc(C(=O)N(C)C)cc1)=O N1(C(C2=NN(C)C(=O)CC2)=O)CC2COCC(C1)C2NC(=O)C=CCO Cn1cc(CC(N2CCC3OCC(=O)NC3C2)=O)c2ccccc2c1=O c1(C(=O)NC2C(C)CN(C(=O)CCC3CCC3)CC2)ccc(P(C)(C)=O)o1 CCCC(CC)CC(=O)N1C2CCC1CC(NC(C1COC(=O)N1)=O)C2 C1(CNC(C2(C)CC(=C)C2)=O)COC(C)(C)CN1C(=O)C(C1CCC1)OC N(C(=NCCCN1CCCC1)NCc1ccc(Cl)nc1)CC(C)(O)C1CCCC1 c1(CCC)c(C(=O)NCC2(F)CN(C(=O)C(C)CO)C2)[nH]c(C)c1C(C)=O N1(C(C2C(NC(Cc3c(C)ncs3)=O)COCC2)=O)CC(O)C(O)C1CO c1(N(C2CCC2)C(N2C(C(C3CCC3)=O)CCCC2)=O)c(Cl)ccc2c1OCO2 C(C(O)C(=O)NCc1cc(C(=O)NCCC2(C)CC2)cs1)SC C(CCOC)(C(=O)N1CCOC(CC(=O)OC)C1)NC(C1C(CC)CCO1)=O C#CCCCC(=O)NCC(C)(Cn1cccn1)NC(=O)C(C1CC1)SC N1(C(=O)Nc2nc(OC(F)F)ccc2Cl)CC(=O)NC2(CC2)C1 c1(C(=O)NCC(CN(C)C(c2c[nH]nc2C(C)(C)C)=O)O)ccc2nn[nH]c2n1 C(=O)(C(C)(C)S(C)(=O)=O)N(C1CN(C(C(n2ccc(C3CC3)n2)C)=O)C(C)C1)C c1(CN(C(C)CCO)C)cncc(CNC(c2cc(CO)[nH]n2)=O)c1 c1(C(C(=O)NC2C(NC(c3onc(CC)n3)=O)CC2)OC)cccc(Cl)c1 n1(CC(=O)NCC2CC(NC(C3CC3F)=O)CO2)cnc2ccccc2c1=O N1(C(c2cc(C(C)=O)oc2C)=O)CCOCC12COCCN(C(=O)C(C)OC)C2 CC1CCC(CC(=O)NC(CNC(c2cnoc2-c2ccoc2)=O)C2CC2)CC1 c1(CNCCCCN2CCCC(NC(C)=O)C2)nc(O)c2c(C)c(C)sc2n1 C(c1cc(F)c(F)c(F)c1)=CC(=O)NC(C(C)C)CCNC(C1CN(C)C1)=O c1(C(=O)NC2(CCNC(c3ccn(CCC)n3)=O)CCC2)cc(Cl)ccn1 C1(C(=O)NCCCCC(=O)NC)CC(F)CN(C(=O)C=CC2CCCCC2)C1 C1(CC)CCCC1N=c1cc[nH]c(=NCCCc2nncs2)[nH]1 c1(C(=O)NC2C(CNC(c3ccc(C)nc3N)=O)CC2)nc2ccccc2[nH]1 Nc1ccnc(C(=O)NCC2C3CN(C(=O)CSc4ccc(O)cc4)CC23)c1 Cc1nc(Cl)ccc1CC(=O)NC1CCC(C)N(C(c2sccc2F)=O)C1 c1(C(N2CC(O)(C(C)NC(CCNC(C)=O)=O)C2)=O)c(C)noc1C(F)(F)F C(=O)(CCC(C)=O)N(C(CNC(C(CC)C1CCC(=O)N1)=O)C)C Cn1nc(C(N2CC(CC(=O)NCCSCS(C)(=O)=O)C2)=O)cc1C(N)=O Cc1cc(C(=O)NC(C)CC(=O)N(C2CC(C)(C)C2)C)n(C)n1 c1(C(N(CCCNC(=O)COc2ccsc2)C(C)C)=O)cc2ccccc2nn1 c1(CC)n[nH]c(CC)n1.c12ccc(s1)N(CC1CCCC1)C2C(=O)NC(C)(C)CC N1(C(=O)COCc2nc[nH]n2)CCC(F)(C(=O)NCCCC2CCOC2)C1 c1(OC)cc2c(OC)c3c1CCN(CC3)C2.c1(CN)ccc(SC)cc1 Cc1nc(C(C)(F)F)ccc1C(N1CCCCC(NC(c2coc(Cl)n2)=O)C1)=O CCC(C)C(O)CC(=O)NCC(C(=O)NC(c1scnc1C)C)C(C)C C(N=c1[nH]c(NC2CSCC2C)nc2c1CSC2)c1cc(C)c(CO)cc1 c1(C(N2CC(SC)C(NC(=O)C=C(C)C(F)F)C2)=O)cc(C)c2nc(C)cn2c1 C1(NC(C(C)C)=O)CCCCN(C(c2n[nH]c(C3CC3)n2)=O)C1 N1(C(c2ccc(C)[nH]2)=O)CCCCC2(CCN(C(=O)C(O)C(C)C)C2)C1 N1(C(c2ccc(C)cc2C)=O)CC2CN(C(C3COCC3(C)C)=O)CCC12 CC1CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(c1cc(CO)ccn1)=O N12CC3C(C3C1)CNc1c[nH]c(c1)C2=O.c1(CN(C)C)cc(CO)on1 N1(C(C2(CCC=C)CCCC2)=O)CCN(CCCNC(=O)C(=O)NC2CC2)CC1 c1(C(C)=O)cn(C)nc1C(=O)N(CC(C)N(C(=O)C(C)NC(N)=O)C)C c1(CCC(=O)NC(C2CN(C(=O)Cc3ccco3)CCO2)C)nc2ncccn2n1 C12(CC)CN(C(c3ccc(C)n3C)=O)C(CNC(C3CCC(F)(F)C3)=O)(C1)C2 C(C)(C(=O)NNC(=O)c1ccncc1)n1cc(-c2cccc(C(=O)OC)c2)nn1 C1(NC(c2ccn(CC)n2)=O)CN(C(c2cnc(C(C)O)s2)=O)CC1N=[N+]=[N-] C1(COCC(=O)N(C)CC2C=CCCC2)CCCN1C(=O)CSC1CCCC1 C1(CNC(c2cc(CC)on2)=O)CCN(C(C2CCCN2C(=O)NC)=O)C12CC2 c1(C(=O)NC2CC3(C2)CN(C(c2cncs2)=O)C3)c(O)cc(=O)n2c1CCCC2 c1(C(=O)NC2C(NC(CC(CC)OC)=O)C2)cc(=O)c2cc(Cl)ccc2[nH]1 C1(C(=O)NCC(CNC(C2(CCOC)CCC2)=O)OC)CC12CC(C)(C)C2 C(=O)(C(C(C)C)NCCC(C)(O)C1CC1)NCCC(=O)OCC C(=O)(C1c2c[nH]nc2CN1C(C1CCC(=C)CC1)=O)NCC=C N1(C(CN(CCC#C)C)=O)CC2(C(N3CCCCC3CCO)=O)CC1CO2 C1(CC(=O)NCCC(C(=O)OC)C)CCCCN(C(C2(Cl)CCC2)=O)C1 C1(c2n(C)ncc2)C(C(=O)NCC#CCCO)CCC(=O)N1C1CC1 CC1(C)CC2CN(C1)C(=O)C=CC2.c1(NC(C(=O)NCCC(N)=O)=O)ccccc1 C1(CCCC)(C(N2CC(O)(CCNC(c3cnoc3C(C)C)=O)C2)=O)CCCC1 C1(C2CC2)(C(=O)NCC(C2CCCC2)NC(C(C)N2CCC2)=O)CC1 c1(OCC=C)ccc(C(N2CC(NC(c3oncc3CC)=O)CC2C)=O)cc1 C1(CNC(C(c2ccco2)NC(c2c(C)n(C)cc2)=O)=O)CCCC12CCC2 c1(CC)n[nH]c(=NC2CC(NC(c3ccccc3NC(N)=O)=O)C2)o1 C1(CNC(CCC=C)=O)CC2(CCN(C(c3cc(C(C)(F)F)n[nH]3)=O)CC2)CO1 CN1CCCC(c2cn(CCCN(C(c3c(Br)n[nH]c3Br)=O)C3CC3)nn2)C1 c1(CC(N2CC(CCNC(C3(C)CC(C)OCC3)=O)C2)=O)cc2ccccc2s1 CC1CCN(C(c2cccc(CF)c2)=O)CC1CNC(=O)C1=CCOC1 C12(C(=O)NC3CCC(NC(Cc4c(C)con4)=O)CC3)CC3CC(C(=O)N1)C2C3 c1(C(N2C(CNC(c3cc(-c4ccccc4)no3)=O)CC2)=O)cc(O)nc(O)n1 N1(C(c2c(CC)nns2)=O)CCC(N(C)C(c2cccc(F)c2Cl)=O)C(C)C1 C1(C)(CNC(CSCC)=O)CCCN(C(c2cncc(C3CCCCC3)c2)=O)C1 N1(c2nnc(C)cn2)Cc2ccccc2C(COC)C1.C1(C(=O)N(C)C)CN(S(C)(=O)=O)C1 c1(CSC)nc(-c2cn(C(C)(C)C)nn2)n(-c2ccccc2C)n1 Cc1ccc(NC2CC2)c(C(=O)NCC(C)N(C)C(C2CC3C(C2)C3(C)C)=O)c1 C1(n2cnnn2)(CNC(=O)OC(C)(C)C)CCCCC1.c12conc1NC2 N1(C(c2n(C)ccc2)=O)CCN(C(c2scnc2C2CC2)=O)CC(C)(C)C1 C1(C)(CC(=O)N(CC(=O)NCCC)C)CCN(C(C2(Cl)CC2)=O)C1 N1(C(C2CN(C(=O)NC)C2)=O)CCC(NC(C2CCCC(C)C2C)=O)C(O)C1 C=CCC(N=c1nc2c(cnn2C)c(N(C)CC2CC2(C)C)[nH]1)c1ccccc1 C(=O)(CC(O)CCSC)NCC1CCC(NC(c2cc(OCC)ncc2)=O)CC1 c1(C(N(C(CCNC(C(CCC)(C)O)=O)C)C)=O)cc2c(cc1Br)CCN2 C1(C2CC2)(C(N2CCC(NC(C3OCCN(CC)C3)=O)C2)=O)CC=CC1 N1(C(c2cc(C)c(Cl)s2)=O)CCC(CNC(C2CC(N(C)C)C2)=O)C12CC2 N1(C(c2n(COC)ncc2)=O)CCCC1C1CCCN1C(c1c(Cl)n[nH]c1C)=O Cc1oc(Cl)nc1C(N1CCC(C)(CNC(c2cncc(CO)c2)=O)C1)=O C(=O)(CC1=NN(C)C(=O)C1)NCC(C)NC(=O)Cc1ccc(F)cc1[N+](=O)[O-] N1(C(C=C(C)c2ccsc2)=O)CC(NC(c2cnsc2)=O)CC(C)C1 CC(C)C(CCC(=O)NC(C1(O)CCCCC1)C)NC(c1ccc(F)cn1)=O C1(C(=O)NC2CN(C(C3CCC=CCC3)=O)C2)CC2CCCC(C1)C2 C(=O)(C1=CCSC1)NC(c1n(C)ncc1)C(=O)NCC1(C)CC2CC2C1 c1(NC(C(CCC#C)NC(=O)CC2CCCOCC2)=O)ccc2nncn2c1 c1(C(=O)NCC(C)NC(C(CCCC)c2ccccc2)=O)cccc2[nH]ncc12 CC1CCCC=C1C(=O)NCC1CC(F)CN1C(=O)CCc1ccnc(Cl)c1 c1(CC(C)C(=O)N2CCC(CN(C(=O)CC3(C)CC3)C)C2)ccc(F)cc1 C(=O)(C1=NOC2(CCN(S(=O)(=O)c3cc(Br)c(F)cc3F)C2)C1)NCCCCC C(N=c1[nH]c(=NCCNS(=O)(=O)C(F)F)[nH]c2c1SCC2)C1CC(OC)C1(C)C N1(C(c2c(CC)nco2)=O)CCOC2(CCCN(C(=O)CCn3ccnc3)C2)C1 c1(C(N(CCCNC(c2[nH]cc(CC)c2)=O)C)=O)oc2ccccc2c1Cl C(=O)(C(F)C(=O)NCC(C)N(C)C(c1ccccc1F)=O)OCC C1(C(C(=O)NCC(CNC(=O)C(F)(F)c2ccncc2)OC)C)CCCCCC1 C1(NC(c2cc(C)cc(F)c2)=O)CN(C(=O)C(C)CCO)CC2(CC2)C1 CN1CC(NC(=O)CCN(C(C23CC(C#N)(C2)C3)=O)C2CC2)C2(CC2)C1 c1(C(N2CC(O)CC(NC(CNC(CCC)=O)=O)C2)=O)cc2c(n1C)CCOC2 C12(CNC(c3ccc(C(F)(F)F)o3)=O)CC1CN(C(c1ccnc(S)c1)=O)C2 c1(C(=O)OCC)nc(C(N2CCC(CNC(C3CC(C)(C)C3)=O)C2)=O)c(C)s1 C1(C(N2C3CC(CNC(=O)CCC4CC4)C2CC3)=O)COc2ccccc2C1 N1(C(C2=C(C)OCC2)=O)CCC2(CC1)COC(CNC(C1CCCSC1)=O)C2 CCCCCCOCCCN(C)CC1CCSC1.C(=O)(C(C)CSC)N c1(CSCC)ccccc1C(=O)NCC12CC1CN(C(C1CCN(C)C1=O)=O)C2 Cc1cncc(C(=O)NC2CC(C(F)C(N3CCCC(CF)C3)=O)C2)c1 C1(N(C)C(C23CC2COC3(C)C)=O)CN(C(=O)CCc2csc(=N)[nH]2)CC1(C)C CC(CC(C)(F)F)C(=O)NCC1(CNC(c2cc3ncccc3[nH]2)=O)CCC1 Cc1scc(C(=O)NC2(CCC(=O)NC(C)C(O)C(F)F)CCCC2)c1C N1(CCC2CCC(n3cc(CCNC(C)=O)nn3)C2)CCC2(CCCCO2)C1 C1(CN(C(=O)CSc2nnnn2C)C)CCN(C(c2csc(C(F)(F)F)c2)=O)C1 C12(NC(c3cc(CCCC)oc3C)=O)CCC1CN(C(c1ncsc1C)=O)C2 C1(C(N)=O)CCN(CC(N2CCCCC2CNC)=O)CC1.C1(C(=O)OC)CC1Cl N1(C(C2(C)CCCC2)=O)CCC2(CCCC2C(=O)Nc2nnc(C(C)(C)C)o2)C1 C1(NS(C(C)C)(=O)=O)OCC2CN(C(=O)Cc3ccc([N+](=O)[O-])[nH]3)CCC12 c1(C(=O)NC2CCCN(C(c3nc(C(C)=O)sc3)=O)C2C)cc2ccncc2s1 N1(C(C)=O)CCCCC1C(=O)NCCN(C(=O)C(O)c1ccco1)C(C)C CC1(NC(c2scnc2C(F)F)=O)CCC(NC(C2(C)CCOCC2)=O)CC1 c1(OC)cccc2c(C(=O)NC(C)CN(C(=O)CCc3ccoc3)C)coc12 Cc1cccnc1CC(=O)N(CCCCNC(C1CC2CC1CO2)=O)C c1(OC)ccc(CNCCC2=CCCCC2)c(F)c1Cl C1(C(=O)NC2C(CNC(c3nc(OCC)sn3)=O)COC2)CCc2nn[nH]c2C1 CC1CN=C(N2CCN(C(c3cccc(Cl)c3Cl)C(=O)NC(C)(C)C)CC2)S1 C12(CNC(C(C)OCCCC)=O)CCC(CC1)N2C(c1sc(O)nc1C)=O Cc1c(C#N)c(N2CC3CCCC(NC(C4CC4F)=O)C3C2)nc2ccccc12 C12(C(=O)NCC(CNC(C(C)CCc3ccccc3F)=O)C)CCCC1CCC2 N1(C(CC(C)N(C(CN(C)CC)=O)C)=O)CC(C)(C)OCC1C C1(CNC(CNS(C)(=O)=O)=O)C2CCCC1N(C(=O)CN1C(=O)CCC1=O)C2 CC(C)(C)C(O)CN1CCCC1c1ccc(Br)cc1 c1(CCC(=O)NC(C2(O)CN(C(=O)COCc3nccs3)C2)C)ccccc1 CC1CN2CCN1CC2C(=O)N(CCCCNC(=O)C1=CC2CCCC12)C C1(C(=O)Nc2nccnc2C)(NC(C2CCN(CCC)C2)=O)CCCC1C N1(C(c2ccc(OCCOC)cc2)=O)CCC2CC1CN(C(C1(C#N)CC1)=O)C2 C1(NC(c2c(CC)c(C)sc2)=O)CC2CC1CN2C(=O)CCC1OCCO1 S(=O)(=O)(c1ccc(NC2CCOC(c3ccnn3C)C2)c(Br)c1)NCC(=C)F N1(CC(C)C)CCC(C(N2CCC(NC(C3(C4CC4)CC3)=O)C2)=O)CC1 C1(C(=O)NCC(CC)C#N)CCN(C(C2CC(C)(C)CO2)=O)CC1 N1(C(CCCOC(C)C)=O)CCC(C(C)NC(=O)CC2(N(C)C)COC2)CC1 c1(C(=O)NCC(CNC(CC(CC)OC)=O)(C)O)cnn2cccc(C)c12 C(c1ccc(F)c(F)c1)=CC(N1CC(OCCNC(C=C2CCC(C)C2)=O)C1)=O Cc1cc(N2CCC(CC(F)F)CC2)ncc1S(=O)(=O)NC(CO)C1CCC1 Cc1ccc2nc(C)cc(C(N3CCC(O)(CNC(=O)C(O)C(C)C)C3)=O)c2c1 c1(OC)n[nH]c(C(=O)NC2CC(NC(=O)Cc3cncc(C)c3)C(O)C2)c1Cl c1(-c2c(C)cc(C(=O)OC)c(C)c2)cnn2c1CN(Cc1cnc(Cl)nc1)CC2 c1(SCC(=O)NCC(C)N(C(C=CC(C)C)=O)C)n[nH]c(=N)s1 N1(C(CC=C(C)C)=O)CCC(C(=O)NCCC2(C)CCOCC2)C1C1CC1 C=CC(CCC)CC(=O)NCC(CC)NC(=O)CNC(c1cc(C)nn1C)=O CC1(C)CC1(C)NC(c1c[nH]nc1CNC(=O)C(O)C1CCCC1)=O CC1CSCCCN1C(=O)C(CC1CCOCC1)NC(c1cc2n(n1)CCO2)=O Cc1cnc(N2CCC(NC(c3coc(C(N)=O)c3)=O)C(O)C2)nc1C c1(C(=O)NCC(CNC(C2CC(CC)OCC2)=O)C)cccc2nonc12 N1(C(CC(C(C)C)O)=O)CCC(C2CCOCC2)(CNC(c2ccoc2Cl)=O)C1 c1(N2CC(F)CC(NC(Cc3c(C)n[nH]c3C)=O)C2)ncnc2sccc12 N1(C(C2(C)CN(C(C3CCC(CC)CC3)=O)C2)=O)CC(C)(COC)CC1(C)C Cc1c(C(=O)NCC2CCCN(C(=O)C=CCO)CC2)cccc1O c1(C(N2CCN(CC(N3C(C)CCCC3)=O)CC2)=O)csc2nnsc12 Cc1nn[nH]c1C(=O)NC1CC(NC(C2(c3ccccc3)CC(C)C2)=O)C1 C#CC1(F)CCN(C(=O)NC(c2csc(NC(C)=O)n2)C)CC1 C1(C(=O)NC)CCN(C(=O)CC(C2CC2)NC(c2cnc(O)n2CC)=O)C1C C1(C(=O)N(CC(C)OC)C)(NC(c2c(CC)[nH]cc2)=O)CC(F)(F)C1 CC#CCC(C(=O)NCC(F)(F)CC1CC1)NC(c1ccoc1C)=O c1(C(N(CCC(=O)NC(C)CCC2CC2)CC=C)=O)ccoc1CC c1(OC)nc(C(=O)NCC2(NC(C3CCN3C)=O)CC2)sc1C Cn1nc(CNC(C2(NC(=O)C=Cc3cc[nH]c3)CCSC2)=O)n(C)c1=O c1(C(=O)NCC(CC)(C)NC(c2nonc2N)=O)cc(C)nc(O)n1 N1(C(c2c(Cl)ccc(C)c2)C(=O)NC2(C)CC2)CCOC2COCC2C1 Cc1ccc(C(N2CCCC(CN(C(=O)CCc3ccccc3)C)C2)=O)c(C)c1 n1(C(C)C(F)(F)F)nc(-c2cncnc2)nc1C(N)CCC#N CC(CC(=O)N(C)CCC1CCN(C(C2CCCC2C)=O)CC1)CC(F)(F)F c1(CNCC2(C#C)CC2)cn2ccccc2n1 c1(C(=O)NC2(C)CN(C(=O)COC3CCCCCC3)C2)cccc(CC#N)c1 Cc1cccc2c1OC(C(N1CCC(CCNC(C3(O)CC(F)(F)C3)=O)C1)=O)C2 c1(C(=O)OC)cc(OC)cc(C(=O)NC2CN(C(=O)C(N)=O)CCC2F)n1 n1(CC)nc(C)c(NC(=O)COCCNC(=O)CC2COCCO2)c1C c1(NC(c2csc(-c3ccnc(C4CC4)c3)n2)=O)cc(F)c(O)cc1Cl C(c1ccccc1)=CCC(N1CCC(C(=O)NCC2(F)CCC(O)C2)CC1)=O c1(C(N2CCC(C(N(C(C(=O)NC)C)C)=O)C2)=O)cnc(C)[nH]c1=N Cc1sc(S(N)(=O)=O)cc1C(=O)NC(CNC(=O)CC(=O)NC1CC1)C1CCC1 c1(C(N(CCCNC(=O)C=Cc2cc[nH]n2)C)=O)cc(Cl)cc(Cl)c1F CC1(C)C(C(=O)NCC(C)(C)C(C)(C)O)CCN1C(c1ccc(CO)cn1)=O C=CC1CN(C(C2CN(C(c3nc(O)sc3C)=O)CC2CC)=O)CCO1 c1(CC)ccc2c(CC(=O)NC3C4CN(C(c5csnc5C)=O)CC34)coc2c1 c1(C(=O)NC2CC(CNC(C(CC=C)C)=O)C2)cccc(O)c1[N+](=O)[O-] C1(NC(c2cncc(C(F)F)c2)=O)CN(C(=O)C(Cl)=CCl)CCC12CCOCC2 C1(NC(c2c(C(C)C)ncs2)=O)CCOC(CNC(C2CCCN2C=O)=O)C1 C=Cn1cc(C(C(=O)NCc2ccccc2Br)N(C)CC2CCCO2)cn1 c1(C(N2CC(OC)CC(NC(C(C(=C)C)(C)C)=O)C2)=O)sccc1S(N)(=O)=O c1(C(N2CC(c3cn(-c4ccccc4I)nn3)C(O)C2)=O)cc2cnccn2c1 C1(COC)(CNC(=O)CN(C(=O)COCC(C)(C)C)C2CC2)CCC1 C(=O)(CC(C(F)(F)F)n1cccn1)N(CCC)CCNC(=O)Cc1nc(C)cs1 CCC(C)(C(=O)NC(C)C(CO)NC(=O)C(C)NC=O)OC N1(C(CCCNC(C)=O)=O)CCC(C)(NC(c2cc(C#N)on2)=O)C1 C1(C)(C(=O)NC2CC(OCC(=O)NC(c3scc(C)n3)C)C2)CCOCC1 c1(OC)cc(C(N2CCCC(C(N)=O)C2)=O)c(NCc2cnn(CCF)c2)cn1 C1(NC(C2C(CC)CCO2)=O)CC(CO)N(C(=O)CN2CCCNC2=O)C1 C1(CNC(C2C(C)(Br)C2)=O)CC2(CO1)CN(C(c1cc3ccsc3[nH]1)=O)C2 N1(C(CCn2ncn(C)c2=O)=O)CCC(F)(CNC(c2cc(Cl)c[nH]2)=O)CC1 CC1CCC(C(=O)NC(C2CCCCC2)CO)N1C(C12CSCC1C2)=O C=C(C)CC(C(=O)NCC(CC)N(C(=O)CC1(OC)CCCCC1)C)OC C=C1CCN(C)C(C(=O)OC)C1.c1(CCOC)ccc(OCF)c(F)c1 Cc1nc2c([nH]1)CC(C(=O)NC1CC1CNC(c1cc3ncccc3o1)=O)CC2 C1(O)(C(C)NC(=O)C=Cc2ccc(F)nc2)CCN(C(=O)CCOC2CC2)CC1 C1(=CCC)CCN(CC2C=CCN2C(=O)CC2COCCO2)C1 Cc1sc(=O)n(CCC(=O)N(CCNC(C2CCCC2)=O)CC2CC2)c1C Cc1ccnc2nc(C(N3CCC(O)(CNC(C4CC5CCC5C4)=O)C3)=O)nn12 c1(SCC(=O)NCC(C)(C)NC(C(C)C2CCC2)=O)ccccc1Br N1(C(C2OCCN(C(C)C)C2)=O)C2CCC1C(CNC(c1nncn1C)=O)C2 c1(OC)cc(N2CCN(C(C3CCCC(C)(C)C3)=O)CC2C)nc(C)n1 CCC(C)(COC)CNC(=O)C(c1cccnc1)NC(=O)C(C1CCCC1)SC c1(NCc2c([N+](=O)[O-])scc2)ccc(S(=O)(=O)NCC(O)Cn2cccn2)cn1 c1(OC)ccccc1CC(=O)NCC1CN(C(c2ccc(CO)nc2)=O)CC1C c1(CC)cnc(-c2ccc(C(C)NCCc3ccco3)cc2)nc1 C1(CNC(c2c(COC)non2)=O)CCCCC1NC(C1(C)CCCCC1)=O C1(C(=O)NCCCCC#C)CN(C(=O)COCCSC)CCN1C c1(COC)c(Cl)cc(C(=O)NC(C)CC(C)C)cc1Cl C(=O)(C1=Cc2ccccc2C1)NC(CN(C(c1ccoc1C)=O)CC)C c1(OC(C(=O)NCC(CCOC)O)=O)ccc(Cl)c(F)c1COC c1(NCCc2c(F)cccc2Cl)nccc(=NCCc2csc(Br)c2)[nH]1 C(C(COC)C(=O)NCCCCC(=O)NC(C)CCN(C)C)OC C1(CC(C)C)(C(=O)NCCCN(C(c2cc[nH]c2C(C)C)=O)C2CC2)CCCC1 C(C(=O)NC(C)C(=O)NCCN(CCCN(C)C)C)(C(C)C)OC C(C1=NOC2CCCC12)NC(Cn1cc(CNC(CC(CC)OC)=O)nn1)=O c1(C(C)C)cc(C(=O)NC2CCCC2NC(=O)C(C)C(C)(C)O)ccc1F c1(C(=O)NC(C)(CNC(c2cnco2)=O)Cn2cccn2)ccc2ccsc2c1 c1(CC(=O)NC2CC(NC(=O)C3=CCCS3)C2)ccc2c(c1)OCO2 CC1(C)CCC(C(=O)NC2CC(O)C2)(NC(C2CCC(=O)O2)=O)C1 C1(CNC(CCN(C(C2(C#C)CC2)=O)C)=O)(CO)CCCO1 CCC(C)(CC)C(=O)N1CC2(CCN2C(c2cc(C(=O)OC)on2)=O)C1 C(C(=O)NC(CO)CCCNC(=O)Cc1ncn2c1CCC2)(C(C)(C)C)N(C)C C1(O)(C(=O)NCC2(F)CCN(C(CC3(C)CC3(F)Cl)=O)CC2)CN2CCC1CC2 C1(CC(=O)NC2CC2)CC(F)(F)C1.C1CCCNC(=O)COCCO1 c1(C(N2CC(N(C(CC(C)SC)=O)C)C2)=O)cccc(CC(F)(F)F)c1 C1(NC(=O)NC2CCC(CCCC)CC2)Cc2cccnc2NC1=O C1(OC)CCCC(NC(=O)C(C2CCCN(C(=O)CSC3CC3)C2)(C)C)C1 C1(NC(C(C)N(C2CC2)CC)=O)CCCCC1NC(=O)Cc1ccccc1 C1(C(=O)OC2CCCC(=O)N2)Cc2nccnc2C1 N1(C(CC(=O)OCC)=O)Cc2n[nH]cc2C1C(=O)N(C(C)C(N)=O)C C1(C)(NC(C2C(C=C)C2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 C(N=c1ccc(Br)c(S(=O)(=O)NCC2CC23CCOCC3)[nH]1)C1CC(=O)NC1 C1(OC)CC(NC(=O)CCc2ncc(F)cn2)CN(C(c2cccc[n+]2[O-])=O)C1 N1(CC(C)NC(C2CCC(CC)O2)=O)CCN(C(=O)C(C)NC(N)=O)CC1 CCC(CC)CCC(=O)NC(COC)CC(=O)NOCCCCF N1(C(C(CC(C)C)C)C(=O)NC2(C)CC2)CCOCC12CCOC2 N1(C(Cn2c(C)cc(C)n2)=O)CCC2CCN(C(=O)CCCOC(C)C)CC12 C(c1ccccc1C)=CCN1CC(NC(C(C=C)c2ccccc2)=O)C(CC)C1 C(=O)(C1=NOC(C)(C)C1)N1CC(N(C(C(CC)C(=O)OC)=O)C)C1 C(C(F)(F)CC(=O)OC)N1C2CCCC2C1C(=O)OC.C(C)(C)(C)OC Cc1ccc(CN2CCCC(CC(=O)NCC3(O)CCCC3)C2)cc1 CCN(CC(C#N)SC)N1CCC(C(=O)OC)(OC)C1 C1(NC(CCC=CC)=O)CCCN(C(c2cc(C)n(C(C)C3CC3)n2)=O)C1C N1(C(C2C(C(C)C)CCO2)=O)CCCCC1CCC(=O)NCC(C)C(=O)N(C)C C(=O)(C1=CCCCC1C)NC1CN(C(c2c(C)nc[nH]2)=O)CC12CC2 c1(CC)c[nH]nc1C(=O)NCC(C)N(C)C(C1(n2ccnc2)CCC1)=O c1(C(N2C(CC(=O)NCc3ccc(O)nn3)CCCC2)=O)nccc2occc12 CCS(=O)(=O)c1cccnc1NC(C1CN(C(=O)CN=c2cc[nH]cc2)C1)=O c1(NC(C)Cc2ccccn2)ccc2c(c1)nc(C(F)(F)F)n2CC1CC1 c1(CC)[nH]ccc1C(=O)NC1CC(C(=O)N(C)CC2(O)CN(C)C2)C1 C1(CCNC(C(C)OCCCC)=O)CSCCN1C(c1snc(Cl)c1Cl)=O C1(O)(CC(=O)NCC(C)(C)OCC(=O)NC2(C(C)C)CC2)CCOCC1 N1(C(C2=C(C)CC2)=O)CC2CN(C(=O)C(C)C(F)(F)F)CC2C1 C(=O)(C(O)CC(F)(F)F)N1CCC(C(C)NC2(CN(C)C)CCCCC2)C1 C1(C(N(CCCC(=O)NCC(COC)C)C)=O)CC(O)C(F)C1 c1(CC(=O)NCC2(O)CC(C(=O)NCC3(OC)CCC3)C2)cc(C)ccc1C C1(NC(C(CNC(CC)=O)(C)C)=O)CCCCCC1C(=O)NC c1(CC)cccc(C(=O)NCC(C(=O)NC(C2CCOC2)C)N(C)C)c1 N1(Cc2cnn(C(C)C)c2F)CCC(O)(CC#N)CC1 CCCC(C(=O)NCC(CC(C)C)NC(C12CCC(CC1=O)C2)=O)C(C)C C(=O)(C(CC(C)C)C(N)=O)N1CCN(C(c2c(C)nc(=N)[nH]c2)=O)CC1C(C)C C(=O)(CC1OCc2ncccc21)NCC(CNC(CCCC(C)=O)=O)C(F)(F)F Cc1cc(C(N2CC(CNC(C3(C)C=CCCC3)=O)C3(CC3)C2)=O)cc(C)c1F C(C(=O)N(C)CCN(C(=O)Cc1cnc(Cl)cc1C)C)(C(F)(F)F)OC(C)=O Cc1ncc2ccc(C(=O)NC(C3CN(C(c4cnsc4)=O)CCO3)C)cn12 C1(NC(COC2(C)CN(C(c3cnn(CCF)c3)=O)C2)=O)CCCC(F)C1 N1(C(C)(C)C)CCCC(CNC(C2CC2(C)C)COC2CCCCC2)C1 CCCCCCCCOCC(=O)NC1COCC1NC(C1CC(=O)OC1(C)C)=O O=C1NCC(C(N2C(C(=O)NC3CN(CC(F)F)C3)CC2C)=O)N1 C1(NC(c2nc(COC)sc2)=O)CC(C)CN(C(c2ccn3c2CCC3)=O)C1 c1(C(=O)NC2CN(C(C34CC(O)C3C4)=O)CC2O)cc(F)c(F)c(F)c1 c1(CC(N2C(CNC(CN(CCOC)C)=O)CC(OC)C2)=O)ccc(C)nc1Cl C(=O)(C(C)(F)C(=O)N1CCCC(N(C)C(c2ccc(C)cc2)=O)C1)OC n1(CC(F)(F)F)nc2nc1-c1c-2cccc1.c1ccccc1.C1CC1Cl Cc1ncc(Cl)cc1C(=O)N(C1CN(C(=O)C(C)(C)c2ccns2)CC1O)C C1(CNC(=O)Cc2cccnc2)CC2CCC(C1)N2C(=O)CN1CCOCC1=O CC(C)(O)C#CC(=O)NCc1cc(C(=O)NCc2nc[nH]n2)co1 C(CC(C)C(C)(C)C)NC(CC(CNC(CCOCCC)=O)C1CCC1)=O c1(SC)cc(C)c(C(=O)NCC2CC(F)(CNC(C3CCCN3N=O)=O)C2)o1 N1(C(c2c(C)scn2)=O)CCN(C(c2c(N)cccc2F)=O)CC1C1CCC1 N1(C(CC=CC)=O)CCN(C(=O)CC(O)C2CCCC2)C(c2cccc(Cl)c2)C1 c1(OC(C2CCNCC2)C)ccc(Cl)cc1S(=O)(=O)NCc1sccc1Cl c1(C(=O)NCCN(C(=O)COC(F)F)C)ccc(Oc2ccc(Cl)cc2)cn1 C=CC1(Cn2nnnc2N2CC3CCCC23)CCCCC1 C12(NC(=O)CSCc3ncc[nH]3)CCCC1CN(C(c1cc3n(n1)CCC3)=O)C2 C1(C(=O)NCCCN(C(=O)CC(c2ccccc2)OC)CC)CCC(C)(C)CC1 Cc1cn2ccc(C(=O)NCC3(F)CC(NC(C4CCCCC4C)=O)C3)cc2n1 N1(C(C(CC)CC)=O)CC2(CCC(CNC(c3cc(Cl)c(Br)c(Cl)c3)=O)O2)C1 c1(NC(C(C)N(C(=O)CCNC(C2C(C)C2(F)F)=O)CCOC)=O)cc(C)nn1C N1(C(C2C(C)CCC2)=O)CCCC1(C)C(N1CCCC1C#N)=O N1(C(C2C(C)C2)=O)CCC(NC(c2ccc([N+](=O)[O-])cc2Cl)=O)C(F)(F)CC1 C(=O)(C(C#N)C(C)(C)C)N(C1CC(C(=O)NCc2cc(C)c(O)nc2)C1)C C(C1CN(C(=O)C2=CCCO2)Cc2ccccc21)NC(C1C(C(C)O)C1)=O Cc1c(F)ccc(C(N2CCC3(C2)CN(C(C2CC(C4CC4)=NO2)=O)C3)=O)c1F C(=O)(C1=CC(O)C(O)C(O)C1)NC(Cc1ccc(CC)cc1)C(=O)OC C1(NC(C(C)OC)=O)(CO)CCCCC1.c1(C(=O)NC)[nH]c(C)nc1C c1(C(=O)NC2CCN(C(c3ccccc3)=O)C23CCC3)ccc2c(c1F)CCC2 C1(C)(CNC(C(C2CCN(C(c3cc(C)c(C)s3)=O)CC2)C)=O)CCN(C)CC1 c1(NC2CCN(C(C(CC(CC)C)C)=O)CC2C)ncnc2onc(C)c12 CCC(CC(=O)NCCCCC(=O)N1CCC(CO)C1)OC c1(OC)nc(Cl)ccc1C(=O)NCC1(C)CN(C(=O)C(O)CCSC)CCO1 C(CN=[N+]=[N-])(C(=O)NCc1ccc(O)c(F)c1)NC(Cc1c(C)ocn1)=O Cc1cc(C)n(CCCC(=O)N2CCC(NC(=O)CC3(CO)CC3)C2)n1 N1(C(CC)=O)CC2CCC1C1CN(C(C3(C#N)CC4CC4C3)=O)CC21 N1(C(c2cc(CC)c(C)cc2)=O)C2CCC1CC(NC(=O)Cc1coc(C)n1)C2 N1(C(c2nc(OC)nc(O)c2)=O)CC(C)(C)CCC1CNC(c1nocc1C)=O c1(C(=O)NC2(SC)CC2)conc1C(C)NC(=O)CC(C1CC1)C1CC1 CC(=O)CC(C)(C)C(=O)NCC1CCCN1C(c1cnn(CCC(C)C)c1C)=O c1(CNC(C(CC(C)C)F)=O)nc2c(s1)CNCC2 c1(C(=O)NCC(C)(C)NC(CC(C)F)=O)nc2ccccc2cc1Cl CC1CCN(CCN)CCC1N(CCC(=O)NCC#N)C N1(C(=O)Nc2nn[nH]n2)CC(N=c2ccnc(C3CCC3)[nH]2)C2(CC2)C1 N1(C(CC2(OC)COC2)=O)CCC2(CC1)CC(NC(=O)C(C)n1cccn1)CO2 c1(C(=O)NC(C2CN(C(c3ccnc(S)c3)=O)C2)C)ccc2c(c1)COCO2 CCN=C(NCc1ccc(OCC)cc1)NCC1CC(=C2CCC2)C1 c1(C(=O)N(CCO)C2CC2)ccc(-c2ccncc2)cc1F CC1CN(C(C2(c3ccccc3F)CC2)=O)CC1CNC(=O)C(C)NC(N)=O C1(CNC(CCNC(N)=O)=O)CN(C(=O)C(O)C(F)F)CCC12CCC2 c1(NC(C(=O)NCCC(C)(C)Cc2ccccc2)=O)c(F)cccc1Cl N1(C(C2OCCN(CC)C2)=O)CC2CCCC2(CNC(=O)C(F)(F)CO)C1 N1(C(c2c(COC)scc2)=O)CCC2(CC(NC(=O)C(Cl)=CCl)CO2)C1 CCC(C(=O)NC(C1CCCN1C(c1cccc(Cl)c1F)=O)C)C(C)C C1(C(=O)NC)CC(C(=O)NCC(CNC(C2(C(C)(C)O)CCC2)=O)(C)O)=NO1 C1(NC(c2cc(COC)oc2C)=O)CN(C(=O)C2=NNC(=O)C2)CC(F)(F)C1 C1(C)(C(=O)NC(CC#C)CC)CCN(C(c2cn(CC=C)nn2)=O)C1 N(C(=NC(C)C)NC(C)CN(C)C1CC1)C1C(C)(OCC)C1 Cc1c(C(=O)NCCCNC(c2ncoc2-c2cccs2)=O)cncc1N C1(CC)CN(C(c2cnc(SC)n2C)C(=O)NCCOC(F)F)CC(C)S1=O n1(C(CNC(=O)OC)C)cc(C2CC(NC(=O)C(C)N(C)C)C2)nn1 N1(C(C(C2CCC(=O)N2)C)=O)CC2(C1)CN(C(c1ccsc1C(F)F)=O)CCO2 c1(C(N2C(C3(O)CN(C(Cc4c(C)ccs4)=O)C3)CCC2)=O)coc2c1COC2 c1(C(N2CC(CCNC(=O)Cc3cocn3)OCC2)=O)ccc(F)c2occc12 c1(NC(C2C(C(N)=O)OCC2)=O)cc(CNC(=O)COC2CCOCC2)ccn1 c1(NC(c2n(CC=C)nnn2)C2(C)CCC2)cccc(C(C)COCC)c1 N1(C(CN(C)C2CC2)=O)C(C(=O)Nc2cccc(O)c2)CCC1C1CC1 C1(C(=O)NC2C(C)CCN(C(C(CC)(C)CC)=O)C2)Cc2ccccc2O1 N1(C(CC2CC(OCC)C2)=O)CCC(NC(C2CC2c2cccnc2)=O)C1CC C#CC1CCC(CNC(c2cc(-n3cc(C(C)(C)CC)nn3)cc(Br)c2)=O)CC1 C1(C(C2CC2c2c(F)cccc2Cl)Nc2n(C)nnn2)Cc2ccc(Br)cc2C1 C(N=c1[nH]c2cccnc2s1)C1(CNC(C(C)OCC#C)=O)CCC1 N1(C(C2CC=CC(n3cc(-c4n(C)cnc4)nn3)C2)=O)CCCC2C=CC12 C(=O)(C(C)C(=O)N(C)CC=CC(N1CC(C)(C)C1C1CC1)=O)OC C1(CCCOC(COC2(C#N)CCC2)=O)CCC2C1C2(F)F C(=O)(CCC(=O)NC(C)CC(C)NC(=O)CCOC1CCOC1)NCCC C(=O)(C(C)(O)CCC)N1CCCC(N(C(Cc2nc(CC)sc2)=O)CCO)C1 C1(CC)CCN2C(C1)C2=O.C(=O)(C1=CCCCC1)NCC1(O)CC2C=CC1C2 c1(C(=O)NCC2N(C(COC)=O)CC(C)CC2)cc(Br)ccc1[N+](=O)[O-] c1(C(N2CC(NC(C3(OC)CCCCC3)=O)C2)=O)c(C)cc(C)cc1O c1(CCNC(=O)CCC2(NC(c3ccon3)=O)CCCC2)ccc(F)cc1 C1(NC(C(=O)Nc2cccc(C(N(CC)CC)=O)c2)=O)C2CCOC2C12CCC2 CCCCCCC(=O)NC(C1CCN(C(c2nocc2CC)=O)C1)C N1(C(CC(C)F)=O)CCC(CNC(=O)Cc2ccncc2Cl)C(C2CC2)C1 CC(C)CC(O)C(=O)NC12CCC(CC1NC(c1ccc(C#N)cc1)=O)C2 C1(CC(=O)NC(C(=O)OC)Cc2[nH]cnc2C)OCCCN1C(=O)OC(C)(C)C C=CCCCC(C(=O)N1CCC(O)(CC)CC1)NC(c1ncccc1C)=O N1(Cc2c(C)cc(C)[nH]2)SC(C)S(=O)(=O)c2ccccc21 C(=O)(C(C)CCCOC)NCC(C)(C)OCCNC(C(CC=C)C)=O C=CCC(C(=O)NCC1C(CNC(C2(COC)C=CCC2)=O)C1(F)F)N(C)C c1(NC(C2(CCNC(C3CC3Cl)=O)CCC2)=O)cccc(CO)n1 Cc1cc(C(=O)NC2CN(C(C3(CO)CC3)=O)CCC2F)c(C)n1C1CCOC1 N(C1CC(C)n2ncnc21)C(C1(CC)CCCC1)=O C12(C(=O)NCCC(Cn3cc(C(COC)(C)O)nn3)F)CCCCC(F)(C1)C2 C(=O)(C(F)CCC(C)C)NC(CCOC)C(=O)NC1(COC(C)C)CC1 C(C(=O)N(C)C)(C(C)O)NC(c1c(C)ccs1)=O.C1CC(=O)NCCO1 C1(CC(=O)NCCCN(C(c2ccn(CCC)n2)=O)C)CCCCC1F CC(CC(=O)NCC(O)CCNC(C1CC=CCC1)=O)NC(N)=O N1(C(c2cnc(OCC)nc2)=O)CCC(C)(C)C1CNC(c1ccnn1CC)=O Cc1cc(C#N)cnc1C(=O)NC1CCN(C(c2n[nH]c(C(C)(C)C)n2)=O)CC1F C1(CNC(C2(CC=C)CCC2)=O)CCN(C(=O)C(C)OCCOC)CC1(F)F Cc1ccc(-n2nc(-c3ccco3)nc2Cn2c(C)csc2=O)cc1 CCCC(C(=O)N1CCC(N(C)CC)C1)NC(=O)COCCC1CCCCC1 N1(C(c2ccc(C(=O)OC)nc2)=O)CCN(C(C2COCC2O)=O)CC1CC#N CCC(O)C(C)C(=O)NCC1CCN(C(c2cccn2C2CCCC2)=O)C1 N1(C(CC2CCCC(NC(COCCCCC)=O)C2)=O)CCC12CC(COC)C2 C(C(=O)NC(=O)CCc1ccc(N(C)C)cc1)(C(C)C)N(C1CCOC1)C(C)C c1(C(N2CCN(C(c3c(Cl)ncc(C)c3)=O)C(C)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 Cc1ccsc1C(=O)N(CC(C)CNC(=O)CSCC1CCCO1)C C1(CNC(CCSC)=O)CC2CC1CN2C(=O)Cc1ccc(F)cc1 CCC(CN(C)C)C(=O)NC(CCSC)C(=O)NCCN=[N+]=[N-] C(=O)(C1CCCc2ncnn21)N1CC2(CN(c3ncnc(CC)c3OC)C2)C1 C1(C(=O)NCCOCCN(C)C(c2cc(C(C)(F)F)n[nH]2)=O)CCC=CCCC1 N1(C(C(C)(C)C2CC2)=O)CCC2CCN(C(C34CC(F)(C3)C4)=O)C2C1 CC(O)CC(=O)N1CC(NC(c2cc(C(F)F)[nH]n2)=O)C1 N1(C(C2CCc3cncn3C2)=O)CCCN(C(C2CCC=CCCC2)=O)CCC1 N1(C(C(CCSC)O)=O)CC2CC(C1)CN(C(c1ccc3nc(O)cn3c1)=O)C2 N1(C(C(C)CN2CCOCC2)=O)CC2CC1C2NC(c1cn(CC(N)=O)nn1)=O C1(CNC(CCC2(C)CC2)=O)CCCCN1C(=O)C(C#N)=CC1CC1 Cc1cccc(C(N2CCCC2C(C)(C)CNC(C2CC23CCOC3)=O)=O)c1F Cc1ncc2n1CC(C(=O)NC(CO)CCCCNC(c1cnn(C)c1)=O)CC2 N1(C(c2cnc(COC(C)(C)C)o2)C(=O)NCC=C)CC2CCCCCC2C1 N1(C(=O)Nc2c(NC(=O)C3CC3)ccc(C)c2)CCS(=O)C(C)(C)C1 c1(C(N(C2CCN(C(CSCCCC)=O)C2)C)=O)nc2ncc(CCO)cn2n1 CC1(C)CC(CNC(c2ncccc2F)=O)CN1C(=O)Cc1c(O)ncnc1O C1(CF)CCCN(Cc2ncc(-c3ccc(Br)cc3)o2)C1 C(=O)(NNC(=O)c1ccc(CN(C(=O)OC(C)(C)C)CCl)cc1)C12CCCCC1C2 CCC(CC)(CCNC(=O)Cc1ccco1)NC(=O)C(c1nc(F)ccc1Cl)C C(=O)(CC1OCCc2sccc21)OCc1nc(CC)on1 C1(C(=O)NC2CC(NC(C3(F)CCOC3)=O)C2)CCN(C2CCSC2)CC1 C1(C(=O)Nc2cc(OC)ncn2)C2C(CN1Cc1cnsn1)C2(C)C c1(OC)nc(C)cc(=NCC(O)CSc2cccc(NC(C)=O)c2)[nH]1 C1(C(=O)NC(COC)CNC(c2sccc2F)=O)CCC2(CCCCC2)C1 c1(NC(=O)NC(C)C)ccc(CNc2cnc(-c3ncccn3)s2)cc1 N1(C(COC(C)C)=O)CCC(C(N2CCC(c3nn[nH]n3)C2)=O)(CF)C1 N1(C(CC2COCC(C)O2)=O)CCCCC(CC(N2CC(N(C)C)C(C)C2)=O)C1 CC1(C)CCC(C(N2CCCC2C2(C(N(C=O)C(C)(C)C)=O)CC2)=O)CO1 c1(C(=O)NCC2CCCN(C(=O)COC3CC3)CC2)cc2c(F)cccc2[nH]1 c1(C(N(CCC(C)NC(c2c(C)cc(O)nn2)=O)C)=O)cc2ccccc2s1 Cc1nc2cnn(C)c2cc1C(=O)NC1(CNC(=O)C(O)C(F)(F)F)CC1 C1(C(N(CCCCO)CCCC)=O)CCN(C(c2c(F)cncc2F)=O)CC1O c1(C(=O)NCC2(CNC(C3CCN(C)CC3)=O)CCC2)ccc([N+](=O)[O-])cn1 C1(NC(COC(C)(C)CNC(c2ccnc(Cl)c2)=O)=O)CCC(N=[N+]=[N-])CC1 c1(C(=O)NC(C)CC2CN(C(C3CC(F)C3)=O)C2)cc(Br)cc(F)c1O CCC(C)CC(=O)NCC1CC(C(N2CC(C)(C)C2C(C)C)=O)C1 C#CC(CC)(CC)NC(=O)C(F)CC1CN(C(=O)C(CC)CC)C1 Cc1ccnnc1C(=O)NC1CC2(C1)CC2C(=O)NCCC(O)C1CCC1 C1(CNC(C(CC)O)=O)CC12CCN(C(c1cccc(CO)n1)=O)CC2 Cc1cc(F)ncc1-c1cn(C2(C(=O)NCCc3ncon3)CC2)nn1 N1(C(C2(F)C(C)OCC2)=O)CCC(C)(NC(C2CC(n3ccnn3)C2)=O)CC1 c1(C(C)NC(C2CC(NC(C(=O)NC)=O)C2)=O)nnnn1C1CC1 N1(C(=O)CSC2CC2)CC2CN(c3cc(=O)n4ccccc4n3)CC(C1)C2(F)F C1(CNC(c2cn(CCC)nc2)=O)C(C)CCN1C(c1ccc(C(C)C)cn1)=O c1(C(=O)OCC=CC)ccnc(C(F)F)c1 c1(C(N2CCC(C3CCCN3C(=O)CC3CC=CC3)C2)=O)coc(Cl)n1 C1(CCNc2cn(CCO)nn2)(CN)CCCC1 c1(C(=O)N(CCO)CCc2ncon2)cnc(C(F)(F)F)cn1 c1(CC(N2CCC(CN(C(C3C(CC)C3)=O)C)C2)=O)nc(C)sc1C c1(C(=O)NCCNC(c2c(C)cccc2)=O)ccc2cccc(C(C)C)c2n1 C12(C(=O)NCCCC(C)NC(C(C)OC)=O)CCCC1C2(F)F N1(C(c2c(C)c[nH]c2)=O)C(C(=O)NCCCNC(N)=O)CCC1C(C)C C(=O)(C#CC1(C)CCCO1)NC12CC(CNC(c3ccc(C(C)C)o3)=O)(OC1)C2 CC1(C)CC1(C#N)C(N1CC(C(N)=O)(CNC(c2ccncc2)=O)C1)=O C1(CNC(C(=O)Nc2c(C)cccc2C(N)=O)=O)(CO)CC12CCOCC2 N1(C(=O)OC(C)(C)C)CCCC(O)C1C(=O)NCC1(CO)CC1 C1(C(=O)NCc2c(C(N(CC(O)C3CC3)C)=O)n(C)nn2)C2CCC(F)(F)C12 c1(C(=O)NCCC(C)N(C(c2c(C)oc(C)c2C)=O)C)cccc2ncn(C)c12 C1(C2(C)CC2)C(=O)N1.c1(NC(C=CCNC(=O)OC(C)(C)C)=O)csnn1 O=C(C1=CC(O)CCC1)NCC1CN(c2nnc(-c3cccnc3)s2)CCO1 C1(C(=O)NC2(CN(C(C(C)NC(C)(C)C)=O)C)CC2)CCc2nncn2C1 C(=O)(C(C)C(F)(F)C(F)F)N1CC2(C(NC(C3C(CC)C3)=O)CCS2)C1 N1(C(C=CC(C)(C)NC(C)=O)=O)CCCCC1CCNC(C1CC1C(C)(C)C)=O n1(CC)cnc(C(=O)NCCCC(C)NC(c2ccoc2Br)=O)c1 C1(C(=O)NC(C)CCNC(=O)CC2CC2)CCCCC(=O)N1 N1(C(c2nc(C(C)OC)sc2)=O)CCC(NC(C2CC3(CCC3)CO2)=O)C(O)C1 S(=O)(=O)(CCC(=O)NCC(=O)NC1CC1)NC(=O)CN1CCSCC1 C(=O)(C1CCCc2scnc21)N1CC2(C(NC(c3c[nH]c(Br)c3)=O)CC2)C1 C(CCN=c1ccnc(NCc2cccc3cn[nH]c23)[nH]1)OC=C C1(C2CCN(c3nccc(C(F)(F)F)n3)C2)(NC(C2CC(C#C)(O)C2)=O)CC1 C12(C(N3CCC(O)(CC)C3)=O)C(NC(=O)Cc3cn(C)nc3C)C3CC1C2C3 N1(C(C=CC(C)(C)SC)=O)CCN(C(c2cc(C)cc(C)n2)=O)CC(O)C1 c1(C(=O)NCCC2CCCN(C(C(C=CC)O)=O)C2)cc2cccc(C)c2s1 C=CCC(C(=O)N1CC(CCNC(=O)C#CC(C)(C)C)C(C)C1)C(C)C C(=O)(C1(C)CCc2ccccc21)N1C(CNC(c2cc(C(C)C)on2)=O)CC1 c1(C(=O)NCc2nc(CNC(c3nn(CC)c(C)c3)=O)sc2)cc([N+](=O)[O-])c[nH]1 C(=O)(C(F)(F)N1CCOCC1)NC(CN(C(COCCCC#C)=O)CC)C CC(C)C(C)CN=C(NCC(C)(C)CN1CCCC(C)C1)NCCN1CCCC1 C(=O)(C(C(C)C)n1cncn1)NCCN(C(=O)Cc1cncnc1)CCOC c1(C(N2CCC(OCCNC(CN(C)C)=O)CC2)=O)ncn2ccccc12 c1(CNC(c2c(C)cnc(F)c2)=O)cnc2cccc(C)n12 C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCC(C(C)(C)C)NC(C=CCCC)=O Cc1ccc(C(=O)NCC2CC2CC(=O)NC(c2nc(C)no2)C)o1 CCCCC(CC(=O)NCC(C)(C)N(C)C)NC(c1cccc2cncn12)=O c1(NC(N(C2CC(C)OC2)Cc2ccccc2)=O)nc(Br)c(Br)cc1Br C1(CC(N2CCC(O)(CCNC(COCCC(C)C)=O)C2)=O)CCCCC12CC2 CC1Cc2cccc(C(N3CCCC3CN(C(=O)C=CC3(C)COC3)C)=O)c2O1 C1(C#N)(CC(=O)N(CCN(C(C2(C)CC2C)=O)CC)CC)CCC1 N1(C(CCc2c(C(C)=O)c(C)[nH]c2)=O)CC2(CN(C(=O)C3CC3)C3CC3)CCC1C2 N(C1CCCc2cn(CN3CCCC3=O)nc21)C(=O)NCc1cc(C(C)C)[nH]n1 c1(OC)ccc(F)cc1CN1CCC(C)(C(=O)Nc2cc(O)ccc2C)C1 C(=O)(C(C)CS(C)(=O)=O)NCC#N.C12CCN(C1)CC(=O)N2CC N1(CC(=O)NC(CC(C)NC(Cc2cc(C(=O)OC)sc2)=O)C)CC(=O)NC1=O CC(C)CS(=O)(=O)CCC(=O)N1CCC(C)C(NC(C2CC(C)OC2C)=O)C1C N1(C(CCCC(=O)N(C(CC)C)CC(C)C)=O)CCN(C(C)=O)CC(O)C1 N1(C(=O)C=CCF)CCC2C(CCN2C(C2CSC3=CC3COCC2)=O)C1 CN=c1nc(C(N2CCC(NC(=O)COCc3cccc(C)c3)C2)=O)cc(C)[nH]1 N1(C(CS(CC)=O)=O)CCC2CN(C(=O)C(C(C)C)c3cccnc3)C2C1 c1(C(CNC(=O)C(C)=C(C)CC)NC(C2(SC)CC2)=O)cccc(F)c1 C1(C(F)(F)F)(CNC(C2C(OC)CC2)=O)CC=CCO1 c1(CN(C(C2N(CCC)CCC2)=O)C)sc(-c2ccc(Cl)cc2)nc1C CCCC(CCC)NC(=O)CCCN(C(=O)COc1ccccc1)C C1(NC(CC2(C)CCCO2)=O)C=CCN(C(C2CC(=O)N(C3CN(C)C3)C2)=O)C1 N1(N(C2CC(C)(NC(=O)CCCOC(C)(C)C)C2)C)CCC(O)(C(N)=O)C1.C=O c1(N2CCC(NC(C(c3ccc(OC)nc3)(F)F)=O)CC2)nc(C)nc(O)c1C CC1(C)CCCN(C(C2(CO)CN(C(=O)CCOCC(F)(F)F)C2)=O)CC1 C1(C(=O)NCc2nn(CC)nc2C)CC(C)(C)CCN1C(=O)CCn1ccnc1 S(=O)(=O)(c1ccccc1)NCC(=O)NCC(CNC(=O)CC1CC2CCC1C2)O c1(OCC(=O)NCCC(C)N(C(=O)CC2CC(=O)NC2=O)C)cncc(Cl)n1 C1(NC(C(c2ccc(C)cc2)C)=O)CCC(C)N(CC2CCCC2C(=O)O)C1 Cc1nc(C2CC2)oc1C(=O)N(CCCNC(c1cn(C(C)C)nn1)=O)C C(=O)(N=c1nc2cc(Cl)ccn2[nH]1)NC1C(C)(C(=O)O)CCCC1 N1(C(CCCC=C)=O)CCN(C)CC1C(N1CCN(C)C(CC)C1)=O N1(C(c2n[nH]c3c2CN(C(n2ccc(C)n2)=O)C3)=O)CCc2ccc(F)cc2C1 c1(CCC(=O)NC(C)CNC(c2n[nH]cc2F)=O)ccc2c(c1)CCO2 N1(C(COCCC(=O)OC)=O)CCC(NC(=O)CC(C)c2ccco2)C12CC2 C#CC1(C(=O)NCCC2(C(=O)NCC3(C)CCCO3)CC2)CCCC1 C(C(O)CC(F)(F)F)ONC(c1oc(C)c(CO)c1)=O c1(COC)nc(Cl)c(C)c(=NCC2CN(C(c3cc(Cl)cn3C)=O)CCC2C)[nH]1 n1(CC#C)cc(NC(c2n[nH]cc2Br)c2nnnn2CCN2CCOCC2)cn1 CC1CC(C(=O)NC2CC(C)(NC(c3ccc(NC(N)=O)cc3)=O)C2)C(C)O1 Cc1ccc(C(N(C(=S)Nc2ccc(Cl)cc2)Cc2ccccc2)COC)cc1 CN1CC(N(C)C(C2CNC(=O)CN2C(c2cn(C)c(=O)n2C)=O)=O)CCC1=O N1(C(C(COC)n2cc(-c3cc(C4CC4)no3)nn2)=O)CCC(C(C)(F)F)CC1 N1(C(c2nc(C)oc2)=O)CCOC2(CCN(C(C3(C)CC3C(F)(F)F)=O)CC2)C1 N1(C(CSCCCCCC)=O)CCC(C(=O)Nc2cc(C(N)=O)co2)(CC)CC1 Cc1n[nH]c(C)c1CCC(=O)NCCCOCCCNC(c1nocc1Cl)=O C1(C(=O)NC2CC(N(C)C(c3ccccc3)C3CSC3)C2)(CC)CCOCC1 C1(O)(CC(=O)N(CCOC)C(C)C2CC2)CCN(C(c2coc(OC)n2)=O)CC1 CCCCCC(O)C(=O)NC(CCC)C(O)C(=O)NCCc1cccnc1F CC1CN2CCCCC2CN1C(=O)NCc1ccc(CC2CCC2)o1 C1(C(=O)NCCC2CC(C(N3CCC(CN=[N+]=[N-])C3)=O)C2)CSCC(=O)N1 N1(C(C2C(=C)C2)=O)CCC(C)(C)C(C(=O)Nc2cc(C#N)ccc2C)C1 c1(NC2CC(C(=O)Nc3cnsc3)C2)ncc2[nH]ccc2n1 C(=O)(C(C(C)(C)C)SC)NCC(CCCC)NC(c1c(OC)csc1)=O c1(C(=O)NCCC(C)N(C(=O)CC2CCCCC2(C)C)C)c(F)ccc(F)c1N C#CCC(C(=O)NCC1CC1C(=O)OC)NC(=O)CCc1ccncn1 c1(CNC(C2CCNC23CCC3)=O)cc(F)ccc1C(F)F CC1CC(N(C)C(c2cncc(CNC(=O)C(C3CCCCC3)O)c2)=O)CCO1 C(=O)(C(C)C(C)(F)F)OCC(N1CCCC(CCCc2ncn(C(C)C)c2)C1)=O CC1=C(C(=O)N2CC(NC(C3CC4C=CC3C43CC3)=O)CC2(C)C)SCCO1 C1(NC(C=C)=O)CS(=O)(=O)N(C)C12CCN(C(C1(C(F)F)CCCO1)=O)CC2 C(=O)(C1CCCn2nccc21)NCC1(OC)CCN(C(C2(F)CCCC2)=O)CC1 CN1N=C(C(=O)NC(CC(=O)NCC2CN3CCC2C3)C(F)F)CCC1=O N1(C(CS(=O)(=O)NC(C)(C)C)=O)CCC2(CCC2)C(NC(c2cc(Cl)c(Cl)s2)=O)C1 c1(SC(=O)CC2CCC3CCC(=O)N23)ccc2nc(C(F)(F)F)sc2c1 c1(C(=O)NCC(C)NC(C2CCCN2C2CC2)=O)cnn2c1OCC2 C1(CNC(C2C(CCC)CCC2)=O)(NC(=O)C(=O)NCC)CCC(F)(F)CC1 C(=O)(C1=CCCN(C(=O)OC(C)(C)C)CC1)N(N1CC(C)CC(C)C1)CC(O)CO C1(c2onc(CCOC)n2)CC(=O)N(C)C1CNc1cnnn1CC CCC(CC1CCCC1)C(=O)N(C)CCNC(c1cnnc(C2CC2)c1)=O CC(C)C(O)C(F)(F)C(=O)N1CCN(C2CCCC2NC(=O)COCCF)CC1 c1(C2C(C(N3CC(CN(C(c4cn(C(C)C)nn4)=O)C)C3)=O)C2)ccccc1F CCC1=NOC(C(=O)NCC(O)CC(=O)N(C)Cc2ccc(C)nc2)C1 N#Cc1ncc(N2CCC(CCNC(c3ccc(Cl)o3)=O)C2)nc1C#N Cc1nccn1CCC(=O)NCC1(O)CC(CNC(c2cnns2)=O)C1 C1(CC(=O)NC2C3CC2N(C(c2cnn4ccsc24)=O)C3)CCC2(CC1)CC2 CCCCCCC(C)CC(=O)NCCOC1CCN(C(C2CCCSS2)=O)C1 c1(OC)ccnc(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2C)c1F c1(CC)nc(N2CCCC(C(=O)Nc3ccc(C)cn3)C2)ncc1Cl c1(C(=O)NC2CCC(NC(C3CN(CC)C(=O)C3)=O)CC2)ccnc2c1CCO2 Cc1cc(=NC(C)CN2CCC(CN(C)C)C2)[nH]c(NC2CCC3CC3C2)n1 C(=O)(C=C1SCC(=O)N1C)N(C)CCN(C(=O)CC1CCC(C(F)(F)F)O1)C N1(C(C(C)NS(CC)(=O)=O)=O)CCC2(C1)CN(c1ncc(C)cn1)C2 Cc1cc2c[nH]nc2cc1C(=O)NCC(C)N(C)C(C1CCn2cncc2C1)=O c1(CNC(C2C=CCN2C(=O)CC2=CCCC2)=O)ccc(F)c(O)c1 Cc1nc(Cl)ccc1C(=O)NC1CCC(NC(c2cnc(Cl)cc2N)=O)C1 Cc1ccc(CN2CCC2(C)C(=O)NC2CCS(=O)(=O)C2)c(F)c1 [N-]=[N+]=NCCCCCC(=O)NCCn1cc(C(=O)NCCC23CC(CO2)C3)nn1 N1(C(c2cnc(C)s2)C(=O)NCc2ccccc2Br)CCCOCC12CCCC2 Cc1cc(C(=O)NC2CC2NC(C2(C)CCCCC2)=O)c2n[nH]cc2c1 S(=O)(=O)(c1ccc(F)cc1)NCCC(C)(C)NC(c1cc(C)nc(SC(C)C)n1)=O N1(C(C)C)C(=O)COCC1C(=O)NCCCCCN(C(=O)CCc1nc[nH]n1)C N1(C(c2ccc(C)nc2)=O)CCCC(NC(c2cc(C3CCCC3)on2)=O)C1C CC1CCC(O)(C(=O)NC2CC3(C(=O)NC4CC(C(N)=O)C4)COC2C3)CC1 c1(C(C)=O)ccc(C(N2CCC(CN(C(=O)CN3CC(C)C3)C)CC2)=O)cc1F c1(OC)c(C(=O)N(C)CCN(C)C(C2CCC(F)C2)=O)[nH]c2ccccc12 C1(C(C)C)CN(C(c2cnc(C(F)F)nc2)=O)CCN1C(=O)CC1CCCO1 C1(Nc2ccc(C(=O)NCC3N(CC)CCC3)cc2)Cc2cc(F)ccc2O1 CCN=c1[nH]c(C(=O)NCC2C(C)CCCN2C(c2cncn(C)c2=O)=O)cs1 c1(OC)cnc(O)c(CNC(=O)CSCc2ccccc2F)c1 C=C1CC2CC1CN2C(CC1CCOC1)C(=O)NC1CCC(CCC)CC1 N1(C(c2cc(F)cc(Br)c2)=O)CC2CC(C1)CN(C(C1(Cl)CC1)=O)C2 CC1(C(=O)NC2CN(C(=O)Cc3ccc(C#N)cc3)C2)CCc2ccccc2C1 C1(CN)CCC2(CO1)CC(C(=O)NCc1sccc1Cl)C2 C1(C(=O)NC(CC)(CNC(c2cc3c(s2)CCC3)=O)CC)Cc2ccccc2O1 N1(c2cc(OC(C)C)ncn2)CCC2(CC1)CC(NC(=O)CN(C)CCO)C2 C(CNC(c1ncc[nH]1)=O)(CNC(C(=O)NCC(c1ccsc1)C)=O)OC CN1C(=O)CC(CNC(C2(NC(c3cn(C)cn3)=O)CC(CO)C2)=O)C1=O Cc1cc(NC(c2c(CNC(c3sccc3C#N)=O)nnn2C)=O)cc(F)c1 N1(C(CCc2n(C)ncc2)=O)CCC(C2CC2)C1C(=O)NCCc1nnc(O)o1 Cc1ccc(Br)c2cc(C(=O)NCc3cncs3)[nH]c12 N1(C(CC(C)(F)F)=O)CC2(NC(C3CC3(C)C(F)F)=O)CCC1CC2 N1(C(CC(C)C2CC2)=O)CCC(F)C(NC(c2ccc(C(N)=O)s2)=O)C1 CC1CCC(C(=O)NCC(=C2CN(C(C3C(NC(N)=O)C3)=O)C2)F)C1 C=CCC(F)(F)C(=O)NC(COC)CC(=O)NC(C)CC(C)C N1(C(=O)C(c2ccccc2)O)CCC12CCCN(S(=O)(=O)c1ccoc1)C2 CCCC(C(=O)NCC1CCCN(C(=O)C=CC(=O)NC2CC2)C1)OCC CC(CC(=O)NC1COCC1C(=O)NCC(=O)NCC1CCCC1)n1ccnc1 Cc1cc(C(=O)NCC2CC2CC(N2CCC(C)(C)C2)=O)c(F)c(Br)c1 CC1(C)CCN(C(=O)C=CCO)CC1CNC(c1coc(C2CCOCC2)n1)=O N1(C(C2CC2c2cccc(O)c2)=O)CC2CCOCC(C2)C1 C(=O)(C(S(C)(=O)=O)N(C)C)N1CCC(n2cc(-c3cccc(C)c3)nn2)C1 c1(C(=O)NCC2CC(NC(C3OCC(C)(C)C3)=O)C2)cncc2cc(Cl)ccc12 C1(NC(C2CC(CCC(=O)NCC(C)OC(F)F)C2)=O)CC2CC1CC2O C(=O)(CCCCC(=O)N1CC2CC2(C(=O)NCc2cccc(Cl)c2)C1)OC Cc1cccc(C(C)C(N2CC3C(NC(c4cn(C5CC5)cn4)=O)C3C2)=O)c1 CC(CC(C)NC(c1n[nH]cc1Br)=O)NC(=O)CSC(=O)N(C)C C1(C)(CCNC(c2ccn(CC)n2)=O)CCN(C(=O)C=CCNC(C)=O)C1 Cc1nc2cc(-c3nc(C(=O)NCC=C(C)C)c(C)s3)ccc2s1 C(=O)(CCCCCN(C)C)N1CCC(C)C1.C(=O)(CCOCCCSC)NCCCO Cn1cnc2c1CN(C(=O)C(O)CCCNC(c1ccc(O)cc1F)=O)CC2 N1(C(c2n[nH]c(C)c2C)=O)CCC2(CC1)CC2C(N1CCS(=O)CC1C)=O C=CCC(C)(CC=C)NC(c1occc1CNC(=O)C=CC1CCCCC1)=O N1(C(c2c(C)csc2C)=O)CCCC2(CCN(C(=O)CC3CCCOC3)C2)C1 c1(C(CNC(C(=O)NCc2n(CCOC)ccn2)=O)C)ccc(F)c(Cl)c1 c1(C(=O)NC2(C)CC(NC(c3cncc(C4CC4)c3)=O)C2)occ2c1CCCC2 c1(C(N2CC(NC(C(CC)c3ccccc3)=O)C2)=O)ccc(NC(C)C)cc1 c1(NC(C2CN(C(CCC)=O)CC(F)C2)=O)cccc2ccncc12 N1(C(C(CC)C)=O)CCC2(CCOCC2)C(NC(=O)Cc2nc(C)sc2Cl)C1 C(N=c1ccc(S(=O)(=O)N2CCC(C)C2C2CC2)c[nH]1)C1(COCC)CCCC1 C1(CNC(C2(F)C(C)C2)=O)CN(C(C2CC(C)(O)C2)=O)CC1O c1(OC)cc(C)ccc1CNCCc1csc(Br)c1 c1(C(N(CCN=[N+]=[N-])C)=O)cc(CNC(=O)C(C)(C)C2CCC2)ccn1 C(C1C(N(C)CCN(CCCC2(C(=O)NC(=O)OCC)CC2)C)C1(C)C)=CC C(CC(CNC(=O)CCC=C(C)C)NC(=O)CCC1CCOC1)OC S(=O)(=O)(c1ccc(N2CCC3(C2)CC(F)(F)C3)c(Br)c1)NC(c1ccns1)C N1(C(C(C(C)C)N(C)C)=O)CC2CCC1CN2C(=O)Cc1ccc(Cl)cc1F C=C(Br)CC(C)(C)C(=O)NC1CCC(N(C(=O)CCc2cc[nH]n2)C)CC1 Cc1nc(NC(=O)NCCCCc2cnn(C)c2)n[nH]1 C1(CNC(C2(CCOC)CCCC2)=O)CCN(C(=O)CCCCO)CCC1(F)F C(CNC(c1cn(C)nn1)=O)(CC(=O)N1CCCC1(C)C(C)(C)C)OC C1(CNC(C2CC(=O)OC2)=O)CN(C(=O)C(=O)NCC(F)(F)F)CC12CC2 C1(CC(=O)NC2CCC(N(C(Cn3c(C)ncc3)=O)C)C2)CCC(=O)CC1 N1(C(=O)OC(C)(C)C)CCC(N=c2nc[nH]c3[nH]c(Br)cc23)C(F)(F)CC1 n1(C(C(N2C3CC(NC(CSC)=O)(C3)C2)=O)C)ccc2ccccc2c1=O N1(C(c2nccc(C#C)c2)=O)CCC(C)N(C(=O)CN2C(=O)CNC2=O)CC1 n1(CC(=O)NC(c2ccccc2)C(C)NC(C2CSC2)=O)c(C)nn(CO)c1=O N1(C(Cc2c(C)scc2)=O)CC2(CCCN(C(C3(NC(N)=O)CC3)=O)C2)C1 C1(C(N(C(C#C)(C)C)C2CC2)=O)C=CCCN1C(=O)Cc1ccco1 c1(OC)cnc(Cl)cc1C(N1CCC(C(C)(C)NC(c2cnoc2C)=O)C1)=O CCC(O)CC(=O)N=c1cc(C2CCCCN2C(c2cc3cnn(C)c3s2)=O)[nH][nH]1 CC1=CCC(C(=O)NCCOC(C)(C)CNC(=O)CCC2CC2CC2CC2)CC1 C1(C(=O)NCC(=O)NCCC(=O)OCC)OCCC1COC C1(C(=O)NCC(COC)NC(c2ncn(CC)n2)=O)CCOCC1(C)C C1(NC(C2CCC(F)(F)CC2)=O)CC2CC(C1)N(c1nncs1)C2 c1(CC(=O)NC(C(=O)NC(CN(C)C)CO)CC2CCC2)ccc(O)cn1 N1(C(CCc2c(C)ncs2)=O)CC(NC(c2cnn(CC3CC3)c2)=O)CC(C)C1 CC1CC(=O)NC(C(=O)NCC23CC(NC(C4(C5CCCO5)CC4)=O)(CO2)C3)C1 CC(C)C(O)C(=O)N1CCC(OCCCn2cc(CCOC(N)=O)nn2)C1 C(=O)(C1=CC(C)(C)C1)NC(CC)CNC(=O)C(CC1CC1)NS(C)(=O)=O C(=O)(CCCCCn1cnnn1)NCC(CCNC(C1N(C(N)=O)CCC1)=O)O C1(C(=O)NCC(F)Cl)(NC(C2C=C(C)CS2)=O)CCN(C)C1 C1(NC(Cc2cccc(CC)c2)=O)CN(C(=O)Cc2cn[nH]c2)CCC1F C1(CNC(CCC(=C)Br)=O)CC(C)CCN1C(c1n[nH]c(CC)c1C)=O CC(O)C(C)C(=O)NC(C)CC(C)NC(C1(C)CCNC1=O)=O C1(CNC(Cc2c(OC)cccc2F)=O)CC12CCN(C(=O)C(C)CF)CC2 Cc1ccc(F)c(CC(=O)NCCCNC(C2COCCC2C)=O)c1 c1(C(=O)NCC23N(C(C4CN(C)C4)=O)CCC2CC3)cncc2c1CCC2 c1(C(=O)NCC2(CNC(C3CCOC3)=O)CC23CCC3)cnc(O)c(F)c1 c1(C(=O)NC2(CO)CN(C(CC3(C)CCC3)=O)C2)cccc2nccn12 N1(C(CN(C(C)=O)C)=O)Cc2occ(C(N3CC(O)CC(C)(C)C3)=O)c2C1 C12(C(=O)NCC(CC(C)C)(C)C)CC3CC1C2C3(F)F n1(C(CC)CC)nc(C(=O)N(CC(O)CNC(=O)CCNC(=O)CO)C)cc1C Cc1ccccc1Oc1nc(CC2CC2)no1.c1(C)ccc(Cl)cc1 C1(NC(CSCC=C)=O)CN(C(c2cc(OC)ncc2Br)=O)CC1(C)C N1(C(c2cccc3nc(C)nn32)=O)CCOC2(CCCN(C(=O)CCCF)C2)C1 c1(CNC(COCC(=O)NC)=O)ccc(C(N2CC(N3CCC3)C2)=O)s1 C=C(C)C(C)(C)C(=O)N(CC(CO)(CO)NC(=O)CNS(=O)(=O)CC)C CC12CCC(CNC(=O)C(C3CCCC3Cn3cc(CO)nn3)C#N)(CO1)C2 O=C(C#CC1CCCCO1)NCC1CCCN1C(c1nn[nH]c1Cl)=O CC1(C)CC(NC(=O)CC2(C)CCN2C(=O)Cc2cc[nH]c2)C(C)(C)O1 Cc1c(C(=O)NCC2C3CC2N(C(=O)C(F)CC2CC2)C3)cnn1C1CC1 C12(NC(C3=NOC(C)(C)C3)=O)CN(C(C3(O)CC(F)(F)C3)=O)CC1CS(=O)(=O)C2 Cc1ncnc2c1CC(C(=O)NCC1CC(CNC(=O)C(=O)NC3CC3)C1)CC2 C1(CCN(C(C)(C)C)C)CCN(C(=O)OC2CCN(Cc3ccon3)C2)C1 c1(COC)ccc(OC)c(OC)c1.C1(NCC(=O)N)CCN(C(=O)C(C)(C)OC)C1 c1(C(=O)NCCCN(C)C(C2CC23CCCOC3)=O)cncc2c1CCCC2 c1(CNC(CCCN(C)C)=O)ccc(CCNC(C2OC3CCC2C3)=O)cc1 CC(C)C(O)(C(=O)NC1CCN(C(=O)C(C2CC2)C2CC2)CC1)C(F)(F)F c1(C(=O)NC2C(CNC(COC)=O)CCC2)ccc(Br)c(Cl)c1 C1(C(=O)NCCN(C)C(c2cocc2C(N)=O)=O)CCCCO1 CCCC(C(=O)N1CCC(C)C(Nc2ccc([N+](=O)[O-])cc2)C1)C(C)C c1(C(=O)NCCC(C(C)C)NC(C2(CC=C)CC2)=O)cc2c(F)c(F)ccc2[nH]1 CCN=C(NCCN1CCCC1)NCc1cc(C)no1.C12CC1C2 C1(C(C)NC(C=CC(CC)C)=O)CCN(C(C2CC2c2cncs2)=O)CC1 c1(C(N(CC(=O)N(CC(C)NC(CN(CC)CC)=O)C)CC)=O)ccsc1 C(=O)(CC1OCCc2ccccc21)N(C(C)C)CCNC(C1CC2(CCC2)C1)=O N1(CC)CC(C(=O)NCC2CCN(C(=O)CCc3cc[nH]n3)CC2C)CCC1=O C(CC(O)C(=O)N1CCN(CCCCCNC(=O)CC2CCC(=O)C2C)CC1)SC C(=O)(C(C)(C)CCC(=O)NC1CC(NC(=O)C(CC2CCC2)OC)C1)OC c1(C(N(C)CC2OCCN(C(CCC#C)=O)C2)=O)cc(F)cc2ccccc12 N1(C(C(c2ccnn2C)C)=O)CCC(NC(c2cc(C3CC3)ns2)=O)C(F)C1 Cc1cc(C)c(C(N2CC(NC(c3nn(C)cc3[N+](=O)[O-])=O)C(O)C2)=O)c(N)c1 C1(NC(C(C)=CC)=O)CC(OC)CN(C(C2(C(F)(F)F)CCCCC2)=O)C1 C1(CNC(C=CCNC(Cn2c(C)ncc2)=O)=O)CCCCN1C c1(CC)nc(C)c(C(=O)NC(C2CCN(C(C3CC(CC(F)F)C3)=O)CC2)C)o1 N1(C(c2onc(COC)n2)=O)CCC(F)(F)C(CNC(=O)C=C(Cl)Cl)C1 C1(C(N(CCCNC(=O)C(C)(C)OC)CC)=O)Cc2cc(Cl)ccc2C(=O)O1 CCCCC(O)CC(=O)N1CCCC(C(N2CCC(C)(COC)C2)=O)CC1 C1(C(N2C(c3n(C)cnc3)CCC2)=O)(CO)CC(F)(F)C1 c1(C(=O)NC(COCC)C(=O)NC2CCCC2(F)F)ncncc1Cl N#Cc1nc(Br)cnc1NC(C1CC1NCc1ccc(Br)[nH]1)=O C1(NC(C(C)OCC#C)=O)CCSC12CN(C(=O)CC1(C)CC1(Cl)Cl)C2 n1(C(C)C)cc(C(N2CC(NC(C3CC(N4CCCCC4)C3)=O)C2)=O)nn1 c1(CC(=O)NC2CN(C(C(CC=CC)C)=O)CC2O)ccc(F)cc1C c1(C(N(C2CCN(C(c3ccc(OC)c(Cl)c3)=O)C2)C)=O)cc2ncccc2[nH]1 C1(N(C(C)C(NC[Si](C)(C)C)=O)Cc2ccccc2)CCCNCCC1 N1(C(C(C(C)C)O)=O)CC2(C)CC1(C(=O)NCc1cc(O)nc(O)n1)C2 N1(C(c2cc(CCC)on2)=O)CC2=C(C1)CN(C(c1ccnc3ccnn13)=O)C2 C#CCCN=C(NCC(C)(C)C(=O)OCC)N1CCC2(CCOCC2)C1 C(c1ccc(C#N)cc1)=CC(=O)NCC1C(NC(c2cn(C)nn2)=O)CCCC1 c12cc(ccc1N)C(=O)OCC(C)n1cc-2nn1.c1(CC)nc(COC)cs1 C=CC1(CC(=O)NC2(CCO)CN(C(=O)C(C)(C)NC(=O)OC)C2)CCC1 c1(OC)cccc(C=CC(=O)NCCc2ccc(Cl)c(C(=O)NCCO)c2)c1 c1(CCCC)ccc(C(=O)Nc2nccc(SC)n2)c(Cl)c1 c1(C(=O)NCC(CN(C(=O)CC(O)c2ccccc2)C)(C)C)ncncc1F C1(C(=O)NC2CCN(C(=O)Cn3ccccc3=O)C2)CCn2ccnc2C1 N1(C(=O)NCCc2cnn(C)n2)CCC2(C1)c1[nH]cnc1CCN2S(C)(=O)=O c1(NC)ccccc1C(=O)NC1CCN(C(=O)CC(C)(C)C2CC2)C1 c1(C(N(C)CCc2nccs2)=O)conc1CNC(=O)C(O)C1CCCC1 CCCCC(C)CCC(=O)NC1(CCCNC(=O)CS(=O)(=O)C(C)C)CC1 C1(CNC(C(C=CC)O)=O)CCC12CCN(C(=O)Cc1cn[nH]c1)CC2 N1(C(c2c(C)ncs2)=O)CC2CC(NC(=O)COc3cccc(F)n3)CC1C2 C1(C(=O)OC)CCCN(CC(=O)NCc2nc(Cl)ccc2Cl)C1=O C1(C)(C(=O)NC(CN(C(c2ccc(Cl)c(Cl)c2)=O)CC)C)CC(C2CC2)=NO1 N1(C(C(CC#C)(C)NC(=O)CC2CC(C(=O)OC)C2)=O)CCC(C)C(F)(F)C1 C(C(COC)CC(=O)N1CC2(C)CC1(C(=O)NCC1CCCCC1(C)C)C2)OC c1(CC)cnn2c1CCC2.C12(COC1)C(=O)NC(C1CC1)CN(C)C2=O C1(CNC(C=C(C)Cl)=O)CCN(c2nnc(Cc3cccc(F)c3)s2)CC1 Cc1cc(F)c(C(=O)NC2CC(CC(=O)N(CC(O)C(F)(F)F)CCO)C2)c(F)c1 c1(-c2nc(NC(Cc3ccn(C)n3)=O)sc2)cn(C)nc1C(N)=O C1(NC(=O)C=Cc2cncc(O)c2)CCN(C(c2cc(Cl)cs2)=O)CCC1CO c1(C(N2CCCC(CN(C(C3CCN(C)C3)=O)C)C2)=O)cc2ccsc2n1C c1(C(=O)NCC2OCCN(C(c3c(C)oc(C(C)C)n3)=O)C2)ccnc(O)c1F C1(CNC(c2cc(CC)n(C)n2)=O)COCCN(C(C2C(F)(F)C23CC3)=O)C1 c1(C(=O)NCC#CC(=O)OC)ccc2c(c1)C(C1CCNCC1)CN2 N1(C(c2nc(C)[nH]n2)=O)C2CCC1CN(C(C1CCCC(F)C1)=O)C2 CN1CCN(C(=O)CN2CCOC2=O)C(CNC(=O)CO)C1 Cc1cc(N)cc(C(=O)NCC2(NC(c3ccsc3C)=O)CCOCC2)c1F CCC(C)CCCC(=O)NC1C=CC(CC(=O)N(CCOC)C(C)C2CC2)C1 C1(NC(C2CC(C)(F)C2)=O)CN(C(c2cc(F)cc(F)c2)=O)CC1C1CC1 CC1(C(=O)NCC(C2CC2)NC(c2cccc(C#N)c2)=O)CC2CCC1O2 c1(C(CF)NC(=O)NC(C(CC)C)CO)cccc2ccccc12 C1(c2n(CCOCC)nnn2)(NCCc2ccccc2Br)CCSC1C C(c1ccccn1)=C(C(=O)NCC(CNC(c1cscc1Cl)=O)OC)C CC(C)CCC(F)C(=O)NC1(C(=O)NCC(c2ccsc2)C)CC(F)C1 CC1=NOC(CC(=O)N(C(C)C(=O)NCc2ccc(C)s2)C)C1 C1(CCNC(Cc2c(C)nc[nH]2)=O)CN(C(=O)Cc2csnc2C)CCCO1 C1(C(=O)NCCCN(C(c2sc(C)cc2C)=O)CC)CN(C)CCO1 Cc1ncnc(N2CC3C(NC(=O)COCc4ccncc4)C3C2)c1C#N C(CCC)(C(=O)NC1CCCC1NC(=O)CSc1ccc(OC)cc1)=CCC C1(N)(C(N2CCCC(C(N(c3ccccc3)C)=O)C2)=O)CC(O)C1(C)C C1(NC(c2n(CC)ncn2)=O)C2CC(O)C1N(C(c1cnc(SC)n1C)=O)C2 c1(CCC(=O)NC(C)CN(C)C(C2CC3(CC3)CO2)=O)cnc2ccccc2c1 N1(C(=O)Cc2ccsc2Cl)CCC2CN(C(c3c(Cl)cncc3Cl)=O)CCC2C1 C1(NC(COC)=O)CN(C(=O)CCN(CCC(C)(C)C)C)CCC1O N(C1COCc2cc(CN(C(=O)CC3CCO3)CCN)ccc21)C(=O)OC(C)(C)C C1(C(=O)NCC(C)CN2CCCC2)CC2(CC2)CN1C(=O)CSC1CCOCC1 C1(n2cc(CNC(C3C(=C)CC3)=O)nn2)CCCN(C(c2cnc(CC)[nH]2)=O)C1 C1(CCC=C)(C(=O)NCCc2ncoc2C)CN(C(c2cccnn2)=O)C1 Cc1nc2cc(C(N3CC4(C3)SCCC4NC(=O)C(C)C3CC3)=O)cnc2[nH]1 C1(C(N2C(C)(C(=O)NCCn3cc(CO)nn3)CCC2)=O)CC2C=CC1CC2 C1(C(=O)NCC2N(C(C3(N=[N+]=[N-])CC3)=O)CC2)CCC2(CC1)CC2 c1(C2CCN(CC(=O)OC)C2)ccc(C)cc1-n1ccc2c(Br)ncn2c1=O c1(C(N2C3C(NC(CC(C)C(F)F)=O)C(C3)C2)=O)cc2ccc(F)cc2cn1 C1(C(=O)NCc2occ(C(=O)NC(c3ccns3)C)n2)CC(=O)NC(C)C1 c1(OC)cc(C(=O)NCC(C(C)C)NC(=O)Cc2cc(C)sc2C)cc(F)n1 N1(C(c2cc(OC)ns2)=O)CCOC(C(C)NC(c2cnc(OC)nc2)=O)C1 C(=O)(C1=CC2CCCCCCC12)Nc1ccncc1.CC1CNC(=O)C(=O)NC1 N1(CC(N2C(CCNC(c3cnc(C)s3)=O)CCC2)=O)CCC(C)CC1 c1(CC)c(C(=O)NC2CC(F)CN(C(c3cc(C4CC4)on3)=O)C2)cccc1F C(C(=O)N1CCC1C1CCC1)(c1ccoc1)NC(CSCCC)=O Cc1nnccc1C(=O)NCCC1CCCN1C(=O)C(C)C(=O)OC(C)(C)C c1(OC)ccc(CC(=O)NCC2(NC(=O)CC(C)c3ccncc3)CC2)cc1F C1(C(=O)NC2(C(=O)NCC3(C#C)CCC3)CC2)CCCC(=O)CC1 CC(CC(C)(F)F)C(=O)NC1(CO)CCN(C(C2(F)CC2)=O)C1 C1(CN(C(c2ccnc(O)c2)=O)CC)CCCCN1C(c1cnc(NC)cn1)=O CC(CC(F)(F)F)C(=O)NC1C2CC3C1C3C2C(N1CCCCC1C1CC1)=O C(=O)(CS(=O)(=O)CCCc1ccccc1)N(C)CC1CN(C(CCC(=C)Cl)=O)C1 N(C1CN(C(=O)C(F)CC2CC2)CCc2ccccc21)C(Cc1nnc(C)s1)=O c1(-c2nc(C3C(NC(=O)C(F)(F)C(F)F)CS3(=O)=O)on2)ccc(O)c(F)c1F C(CCC(C)(C)C)(C(=O)O)NC(C(=O)N(CCC)Cc1ccc(CCC)s1)=O CN(OC1CCCC1)C(=O)C1CC1NC(=O)CC1COCCO1 Cc1cn(CC(=O)N(C(C)CN(C)C(C2(C)CCC(=O)NC2)=O)C)c(=O)nc1O CC1(C)CN(C(C2COC3(CCC3)C2)=O)CC1NC(=O)Cc1c[nH]c(=N)nc1O CC(C)(CNC(=O)C(c1ccoc1)NC(c1cn(C(C)C)cn1)=O)CO CC1NC(=O)CCC1CNC(=O)C(C)N(C(=O)CCCCN(C)C)C C(=O)(CC(O)CCSC)NC(CCCC)CNC(c1ccc(C)cn1)=O C1(C(=O)NCC2=CCN(C(C3C(C#N)C3)=O)CC2)CCCCCC1(F)F Cn1cnc(N2CC(O)(CCNC(C3(C(F)F)CCCC3)=O)C2)c(Br)c1=O CC1CN(C(c2cc(C3(O)COC3)on2)=O)CCC1NC(c1cn(C)nn1)=O C(=O)(C(O)CC[S+](C)C)N1CCC(C)(NC(C2CCC(OC)CC2)=O)C1 c1(N(CC(C)NC(C(C)n2ccnc2)=O)C)nc(Cl)c(C#N)s1 N12CCC(C(C)C1)NC(=O)C1(CC1)C2=O.c1(C(C)C)cccc(CN(C)C)c1 C1(NC(C(CCC=C)NC(=O)Cc2cnn(C)c2)=O)CCn2nnnc2C1 c1(C(C)C)csc(-n2cc(C(C)NC(C3CC3C(=O)NC(C)(C)C)=O)nn2)n1 C#CCCC(C(=O)NCCC#N)N(C(c1cc(Cl)ccc1OC)C(=O)OCC)C Cc1nc(C(=O)NCC(C)(CO)NC(C2CCCCC(=O)N2)=O)ccc1Br CCC(C)(CO)C(=O)NCC1COCCN(C(=O)Cc2cccc(Cl)c2F)C1 c1(NC(CCC(=O)N(C)Cc2csc(CO)n2)=O)ccc(F)c(F)c1 C(c1c(Cl)ccc(Cl)c1Cl)=CC(=O)NCC1CCN(C(=O)CCC2CCC2)C1 c1(C(N(C)CC23CC2Cc2c[nH]nc23)=O)cccc2c1CCS2(=O)=O C#Cc1cc(C(=O)NCC(CC)NC(=O)C(O)C(C)(C)C)cc(O)c1 C(C)(C)(C(=O)N1CCC1CNC(c1c[nH]c(C(=O)OC)c1)=O)NC(=O)OC c1(C(=O)NC2CC(NC(c3n(C)nc(O)c3)=O)C2)csc2c(F)cc(F)cc12 C1(CNC(=O)Cc2cc[nH]n2)(CO)CCN(C(C2CC(O)C2)=O)CC1 C1(C(=O)NC2(C)CCC(NC(CC=CC)=O)CC2)Cc2cccnc2C1 C(CCSC)(C(=O)N(C)CCNC(=O)C(C(C)C)SC)OC CC(CC(=O)N1CCC(CBr)(NC(=O)Cc2ccnc(C(N)=O)c2)C1)C(C)(C)C CCC(C)CN=c1[nH]c(N2CCOC3COCCC23)nc2c1CCCCC2 C(=O)(CCCCCC#N)Nc1cccc(OCC(=O)NCCN2CCC(C)C2)c1 c1(C(N(C(C(=O)NC2C(C)SCC2)(C)C2CC2)C)=O)cn(C)c(=O)cn1 C1(CNC(C(CC2CCOCC2)NC(C(C)SCC)=O)=O)CC2(CC2)C(=O)O1 c1(NC(CC)CC#N)[nH]c(=NC2CCN(Cc3ccnn3C)CC2)nc2scnc12 c1(CC(=O)Nc2cccc(CN(C(C=NOC)=O)C3CC3)c2)ccc2c(c1)COC2 c1(N2CCC(C)C(CNC(=O)Cc3nncn3C)C2)ncc([N+](=O)[O-])cc1Cl N1(C(CCC)=O)CCCC2(CCN(C(=O)C(c3cccc(OC)c3)O)C2)C1 Cc1noc2ncnc(NC3CCN(C(=O)C(N4CCCCCC4)C)C3)c12 C1(C(=O)N(C2CCN(C(=O)C(C)CSC(F)(F)F)CC2)C)(OC)CCOCC1 N1(C(CC2CCC(OC)CC2)=O)CCCC(C)(NC(=O)Cn2cccc2)C1 Cn1nc(C(=O)NC2CCCCN(C(C3CCCC3O)=O)C2)c2cc(F)ccc12 Cc1cc(C(=O)NC(CCOCCO)C(=O)N2CCOCC2C(C)C)cc(C)n1 CN1CCC(C(=O)NCCCCn2cc(C3COC(C)(C)C3)nn2)C1=O C1(NC(c2ccc(OC(C)C)nc2)=O)CCCN(C(c2cnn(C)n2)=O)CC1 CCN=C(NCCSc1ccccc1Br)NC1CCOc2ccccc21 n1(CCCC)nc(C(C)SC)nc1-c1c[nH]ccc1=O Cc1cc(C(=O)N(C2CCN(C(c3cnn(C)n3)=O)C2)C)n(C(C)(C)C)n1 C12(NC(=O)Cn3cncn3)CCN(C(c3cc4ccccn4n3)=O)CCC1C2 c1(C(N(CCCN(C(C(C(C)C)NC(C)=O)=O)C)C)=O)ccc(C#N)c(O)c1 C1(NC(=O)CN2CCCC2CO)CCC(NC(=O)C2=CCCS2)CC1 CON(CCC(=O)NC1CCCCC1N=[N+]=[N-])C(=O)c1cc(Cl)cnn1 c1(NC(C(c2noc(C)n2)N(CC(CC)O)C)=O)ccc(Cn2cccn2)cc1 C(C)(CCC(=O)NCC(c1cccc(Cl)c1)NC(=O)C=C=CC(F)(F)F)OCC C(=O)(CCCS(C)(=O)=O)NC1C2CN(C(C3(COC)CCCCC3)=O)C1C2 c1(OC)ccc(Cl)c(C2(C(=O)NCC(O)CN(C(=O)CC(C)COC)C)CC2)c1 C(=O)(CCCS(C)(=O)=O)N1C(C)CN(C(=O)C(F)(F)C2(O)CCC2)CC1 C1(CNC(c2ccc(C(C)=O)[nH]2)=O)CCCC1NC(c1ccnn1CCF)=O CS(=O)(=O)C1(C(=O)NC2CCC(NC(c3cc(C(F)(F)F)ncn3)=O)C2)CC1 C1(C(N(C)CC2(C)CCCO2)=O)CC(C)(C)CCN1C(=O)Cc1ccsc1 C1(OCC)CCN(C(=O)CC2CCN2C(c2cc(C)sc2C)=O)CC1 C=CC1(CC(=O)N(CC)Cc2ccccn2)CN(C(=O)CC)C1 N=S1(=O)CCC(C(=O)NC2CCCC(NC(c3ccccc3F)=O)C2)CC1 c1(C(=O)NCC(C)N(C)C(C2OC(C)(C)OC2(C)C)=O)ccc2c(n1)COCC2 C1(C(=O)NCCSCCC=C)CN(C(=O)Cc2nocc2CC)CC1(C)C O=C(C1=COc2ccccc2O1)NC1CC(F)(CNC(c2cscn2)=O)C1 Cc1ccc2nc(SCC(=O)NC3CCCC3NC(c3c(CO)cno3)=O)[nH]c2c1 C1(N(C)C(C2COCCOC2)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC12CC2 c1(C(N2CCN(C(C3CC(CCC)OCC3)=O)CC2C)=O)cc2cccnc2[nH]1 N1(C(CN(C(COC)=O)C)=O)CCC(NC(c2cnc(O)n2C)=O)C1C(C)(C)C c1(C(=O)NCC(CSC)NC(CN2CC(CC)C2)=O)ncsc1Br c1(C(=O)NCCC2CN(C(c3cc(F)cc(Br)c3)=O)C2)coc2c1CCCC2 C(C(C(=O)NCCN1CC2CC2C1)NC(=O)C(C1CCCO1)OC)OCC c1(CC(=O)NCC2N(C(C(COC)C)=O)CCCC2C)c[nH]c2cc(C)ccc12 C(=O)(C#CC(C)(C)C)N(CC(=O)N(CCC(F)(F)F)C)C(C)C C(=O)(C(=O)CC(=O)c1ccsc1)N1C(C(C)NC(=O)CN2CCC2)CCCC1 n1(CC(C(C)(C)C)O)nc(-c2cccc(C(F)F)n2)nc1C1COc2ccccc21 N1(C(Cc2c(C)noc2C)=O)CCC2C1CCN2C(c1cc(Cl)ccc1Br)=O c1(C(N(CCC)CCNC(C2CC2(C)C)=O)=O)cc(=O)c2ccccc2[nH]1 C(=O)(C(CO)C(C)(C)C)N(CCC)CCNC(C1(C(=O)NCCF)CCC1)=O CC1CN(C(=O)CC2(C(F)(F)F)CC2)CC1NC(=O)Cn1cc(Br)cn1 CCCCC(O)CC(=O)N1CC=CC1C(N1CC(C)(C#N)C1)=O C1(NC(c2ncn(C)c2)=O)CN(C(C2(C(F)F)CC(F)(F)C2)=O)CCC1O N1(C(CS(CC)=O)=O)CCC2CCCN(C(=O)CC3(N(C)C)CCCC3)C2C1 C1(CCC(=O)N(CCNC(CC2CN(C(C)=O)C2)=O)C2CC2)CC(C)(C)CO1 c1(C(=O)NCCCN(C(C)C)C)cccc(CNC(C2CCCOC2)=O)n1 c1(NC(=O)NC(C)Cc2ccc3c(c2)OCO3)cc(C#N)cc(Cl)n1 C1(CNC(c2ncn3ccccc23)=O)CC2(CCN(C(C3CC3F)=O)CC2)CO1 CCCC(C(=O)NC(C)CN(C)C(C)C)NC(c1cc(CC)sn1)=O C1(C)(CCNC(C(CC=C)OC)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1 c1(C(N2C(CC)C(NC(c3ncc(N)cc3Cl)=O)CC2)=O)cc2c(o1)CCCC2 c1(C(N2C(CNC(=O)COc3ccc(C#N)cc3)CC2)=O)nnn2c1CSCC2 c1(OC)cc(C(=O)NCc2nc(CNC(=O)C=C(Cl)Cl)cs2)n(C)n1 C(CCNC(=O)COc1ccc(C(C)=O)cc1)(C(C)C)N(C(CC(=O)NC)=O)C c1(C(=O)NCC2N(C(CN(C3CC3)CC)=O)CCOC2)cc2c(cn1)COCC2 N1(C(C(C)(F)F)=O)CCC(F)C(NC(C23CC(CO2)C3(C)C)=O)C1 n1(CC(=O)N)cc(CS(C)(=O)=O)nn1.CC(CCC1CC1)n1cccn1 CC1CN(C(=O)CN2CCC(O)CC2)CC1CNC(c1csc(CO)n1)=O CCC(F)(F)CC(=O)NC1CCCN(C(C2CCC2(C)C)=O)C1 c1(CNC(CCN(CC#C)C(C2CCOC(C)C2)=O)=O)ccc(F)c(C)c1 CC1C(C)N(C(c2ns[nH]c2=O)=O)CCN1C(c1nnn2c1CSCC2)=O C#CCCC(O)C(=O)N1CCC(N(C(=O)CC(C)(C)OC)CCC)C1 CC(C)CC(C(=O)NCC1CC(C)CN(C(=O)C(N2CCNC2=O)C)C1)C(C)C N1(C(c2c(Cl)ccc(OC)c2)=O)CCC2(CC1)CC2C(N1CCOC(CO)C1)=O C1(C(=O)NCC2C(C)CCN2C(=O)C(CO)N(C)C)C2CCC3(COC(=O)C13)O2 CCCC(C(=O)NC(CO)C(=O)NCC(N1CCCC1)C)NC(C)=O c1(C(N2CC3C(CNC(C4CC45CCC5)=O)(C3)C2)=O)ccc(F)c2ccncc12 Cc1ccc(C(N2CCC(C)C2CNC(c2ccsn2)=O)=O)cn1 C(=O)(C1Cc2ccc(F)cc21)NC1CCN(C(c2n[nH]c(CC)c2[N+](=O)[O-])=O)C1 N1(C(C(C2CCOCC2)C)=O)CCN(C(c2cc(Cl)ncc2N)=O)CC1C Nc1c(C(=O)NCCN(C(C2CN3CCN2CC3C)=O)C2CC2)cc(Cl)cc1F C1(C(=O)NCC=Cc2c(C)noc2C)CCN(C(=O)C(F)CCC(C)C)C12CCC2 Cc1nc(C(=O)N(C2CCCC2)CCNC(=O)C=C2CCC(C)CC2)c(C)s1 C(N=c1nc(N2CCSC(C(C)C)C2)c2c([nH]1)CCS2)C1CCN(CC)C1 C(C(=O)NCCSCC(=O)NCCCCn1ccnc1)(C1CC1)OC C1(n2cc(CC=C)nn2)CC2CCC1(NC(C1CC(C)=NO1)=O)C2 N1(C(CNC(CC)=O)=O)CCc2nc(CNC(=O)CCOCC3CCC3)sc2C1 C1(NC(C2CC3(CSC3)C2)=O)CN(C(=O)COc2ccccc2)CC2(CC2)C1 c1(N(CC(C)NC(CSc2c(OCC)cccc2)=O)C)ncc2cccnc2n1 C#Cc1cnc(C(N2CCC(O)CC2C(=O)N(C)CCSC)=O)c(C)c1 c1(CC)cnoc1C(=O)NC(C)(C)C(=O)NC(C)CCn1cncn1 c1(C(=O)NCC2(CNC(c3ncn(C)c3)=O)CC23CCC3)cnc2ccnn2c1 N1(C(c2c(CC)nc[nH]2)=O)CC2CCN(C(=O)CN3CCCCCC3=O)CC2C1 Cc1cc(C(=O)NC2CCOC(C(=O)Nc3csnc3C)C2)nc(C)n1 c1(OC)ccc(CNCCN2CCN(C(C3CC3(F)F)=O)CC2)nn1 CCCCC(F)C(=O)NCCCN(C(=O)Cc1ccoc1C)C c1(C(=O)NCCN(C(c2cncc(C)c2)=O)C)cc2c[nH]nc2s1 c1(SC)nccnc1C(N1CCN(C2CCN(C(C3CC(=O)N3)=O)CC2)CC1)=O c1(-c2onc(-c3c(C)ccs3)n2)nn2ccccc2c1Br C=CCC(C)(C)C(=O)N(C1CCCN(Cc2ccc(C(=O)OC)cc2)CC1)C CCCCS(=O)(=O)N(CC(=O)N(CCCN(C)C)C)C.C1(=O)C=C(C)CN1 c1(C(N2CCN(C(=O)CSC3CC3)CC2CCO)=O)cncc([N+](=O)[O-])c1 N1(C(C2CCCCN2C(C2CC(=C3CCC3)C2)=O)=O)CCOCC(O)C1 C(=O)(CCC(C)(C)N(C)C)NC(CCN(C(CCC(=O)NCCC)=O)C)C c1(C(=O)NC(CNC(CC2N(CC)C(=O)CC2)=O)C)cccc2c1C(=O)NC2=O c1(C(=O)NCC2(CCNC(C(CC)(C)C(F)F)=O)CC2)ccc2c(c1)CCN2C S(=O)(=O)(c1ccc(F)cc1F)Nc1cc(S(C)(=O)=O)sc1 C1(NC(c2cnc(CC)s2)=O)CCC2CN(C(=O)Cc3nonc3C)CCC2C1 N1(C(C(CC)(C)CO)=O)CCC2(C=C(C(=O)N(C)CCc3ccncc3)C2)C1 c1(CC(N2C(C)(C)CC(NC(C3CCCCCC3)=O)C2)=O)ccccc1[N+](=O)[O-] Cc1cccc(CCC(=O)N(CCCNC(C2(C)CC=CCC2)=O)C)c1 c1(C(=O)NCC(CNC(C(CCCC)(C)F)=O)C)c[nH]c2ccc(Cl)cc2c1=O n1(CC2(O)CCOC2)c(N(C(c2ccccc2)C2CC(=C)C2)CC)nnc1C c1(C(C)C)ccc(C(=O)N(C2CCCN(C(C3(CO)CC3)=O)C2)CCO)cc1 c1(C(=O)NCC(C(N2CC(O)(COC)C2)=O)OC)ccc(F)c(C)c1 c1(N(C)NCC2N(C(C(C)OCC#C)=O)CCCC2)nc(OC)nc(OC)n1 c1(-c2c(SCC(=O)NC(C(C)C)C(=O)N(C)C)cccc2)ccc(F)cc1Cl C1(NC(=O)CCCC2CC2)CCN(C(=O)COc2ccc(F)cc2Cl)CC1F c1(C(N2CC(F)(CNC(C(C=CC)O)=O)C2)=O)nc(C)sc1Br C1(NC(c2c(N(C)C)cncc2)=O)CCCN(C(C2CCOCC2)=O)CC1 Cc1nc2c(C(=O)NC3CCC(NC(C4CC4(F)Br)=O)CC3)cccc2o1 CC1CCC(C)(C(=O)NCC=C2CCN(C(=O)CC(=O)OC(C)(C)C)CC2)C1 CCCC(C)(O)C(=O)N1CCN(C(c2cc(F)cc(F)c2)=O)CC1C C(C)(CCC(=O)NC(C(=O)NCCCc1n[nH]c(C)n1)C(C)OC)OCC C(C(C)(C)CC1CCC1)NC(C1C(CN(C)C)C1)=O.c1(C(=O)N)cc(C2CC2)no1 Cc1cc(C(=O)NCC2CN(c3nc(C4CCCC4)ns3)CCO2)ncc1F N1(C(C(C2CCN(C(C3C=CCC3)=O)CC2)C)=O)CCN(CCCCF)CC1 C1(c2n(CCSC)nnn2)(NC2C3COCC23)CCCC(F)(F)CC1 C#Cc1ccc(CC(=O)NCC(CC2CC2)C(=O)NC2CC(F)C2O)cc1 C1(C(=O)NCCC)CCCCN1C(=O)NCC1(C)CC1(C)C c1(C(N2CCC(CNC(COCCC(C)C)=O)C23CC3)=O)cnc([N+](=O)[O-])n1C CC1CCCCC1(CNc1ncnc(O)c1Br)NC(=O)Cc1cnn(C)c1 C=Cc1cnn(C)c1C(=O)Nc1cccc(NC(c2nn(CC)nc2C)=O)c1 c1(C(N(CC=C)C2CC2)=O)ccc(CNC(c2n[nH]cc2Cl)=O)nc1 CN1CCC(C(=O)NC(C2CCCCC2)CNC(C2CCC=CCC2)=O)C1=O CCC(C)(CNC(=O)Cc1cccs1)C(C)O.C(=O)(N)O O=C(N=c1cc[nH]cc1Cl)C12CC1CN(Cc1ccc3sccc3c1)C2 C1(CC(=O)N(C2CC(C#N)C2)CC(=O)NCC(C)CO)CCCNC1=O C1(N(C(C(c2ccc(O)cc2)C)=O)C)CCN(C)C1=O c1(OC)ccc(F)c(CN2CCCC2C(=O)NCc2cc(C#N)ccc2Br)c1Br C1(C(=O)NCc2n[nH]c(C)c2C)CN(C(=O)CC(C)c2ccco2)C2(CCC2)C1 CS(=O)(=O)c1sccc1C(=O)NC1CCCN(C(C2C3CC4C(C3=O)C24)=O)CC1 C(=O)(N=c1[nH]onc1C1CCC1)NCCCC(C)O C1(CC(N2CCC(C(=O)NCCO)(CO)C2)=O)CC(=O)c2ccccc2C1 c1(C(=O)NC(C)C(C)NC(C2(C(C)(F)F)CCOCC2)=O)ncc(Cl)cc1F CC1(C)CC(O)CCN(C(c2nc(C3CC3)cs2)C(=O)NCc2cccs2)C1 c1(CN(C(c2coc(C3CCNCC3)n2)=O)CC)cccc(C)c1 N1(C(c2cccc(CC)c2)=O)CCC(N(C)C(c2ocnc2C2CC2)=O)C(C)C1 Cc1c[nH]c(C(=O)NCC2C(C(=O)N(CCC(N)=O)C)C2(C)C)c1 C1(NC(=O)C=C(C2CC2)C2CC2)CCCCCC1NC(C1CC1[N+](=O)[O-])=O CC1=C(C(=O)Nc2cc(C(C)C)c[nH]2)CCC1.C12CCCC(C1)NC1(CC1)CNC2=O C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)C(NC(C(CN)CC(=O)N)=O)CC1 N1(C(C(c2ccc(CNC3(SC)CCCCC3)s2)C)=O)CCC(C(F)(F)F)C(C)C1 C1(C(C2CCN(C(CCc3cnc(C)o3)=O)C2)=O)CCOCC1O.C1C(=O)N1 c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)C(C)CC2)ccc(=O)n2c1CCCC2 c1(C(=O)NC(CNC(C(c2c(C)nn(C)c2)O)=O)C2CC2)sc2nccn2c1C c1(SC)ccc(Cl)cc1NC(c1sccc1I)c1nnnn1C(C)(C)C CCC(F)(F)C(C)(C)C(=O)NCC(C)(C)NC(c1coc(C2CCCCC2)n1)=O CCC(C)(C)CCCC(=O)NC1CCC(NC(c2n[nH]c(C)c2F)=O)C1 C(CC(F)F)(C(=O)NCC(C)(C)CCC=C)NC(CCOCC#C)=O C(=O)(C(C)(O)C(C)C)N1CCCC(CC(NOCCOCC)=O)C1 CCCCC(CNC(C1(F)CC1(Cl)Cl)=O)NC(=O)CC1CC(F)(F)C1 C1(CNC(C(CC)(C)CC)=O)CC2(CCOCC2)CN1C(C12CC1C2)=O c1(SCC)cnoc1C(=O)NC(CO)CN(C(=O)C=CCOCCOC)C C1(O)(CN(C(c2cc(CC)[nH]n2)=O)C)CCCN(C(=O)CC(C)C2CCCC2)C1 C1(C)(C(=O)NC(c2ncc(C)cn2)C)CC(O)CN1C(=O)CN1CCCC1=O C(N=c1ccn(CC(=O)Nc2ccc(C)c(Cl)c2F)c(O)n1)c1cnc(OC)nc1 C#CCC(CC(=O)N(CC(C)CCC)C)NC(=O)CCc1ccccn1 C1(CC)CN(C(c2ncccn2)=O)CCN1C(C1CC(C2CC2)C1)=O C(C(C)(O)CC(=O)NOCC(N1CCC2CCN(C)CC12)=O)OC C1(CNC(c2cn(C)nc2)=O)(CNC(=O)OC(C)(C)C)CC(C)(C)C1 C1(Cn2cc(C3N(C(C(CCC)CCC)=O)CCCC3)nn2)Cc2nnsc2S1 N1(C(CCCC(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCc2cncc(F)c2)C1 N1(C(CCN(C)CC)=O)CCCC(C(C)(C)C(=O)NC2CC3CCC2C3)C1 C1(C(=O)NCC(C)NC(=O)Cc2ccc(F)cc2Cl)C2CCC3(COC(=O)C13)O2 N1(C(C(c2ccc(C(=O)O)o2)C)=O)CCCCC1Cc1cn(CCN(C)C)nn1 c1c2ccc(c(C)c2)c2ccc(c1)s2.c1(S)ccncc1.CCCC=C CC(CC(C)(C)C)C(=O)NCC(O)CNC(c1sc2cncn2c1C)=O C1(CC(=O)NC(CCNC(C(C(C)C)C#N)=O)(C)C)CCC2CC1C2(C)C c1(C(=O)NC2CC(CNC(COCCC#C)=O)C2)ccc(S(=O)C(C)C)cc1 Cc1cnc(C(=O)NC2CC(CNC(c3cnoc3C)=O)C2)cc1Br c1(C(=O)NCC2N(C(c3n(CC=C)ccc3)=O)CC2)cn2c(n1)CCCC2C C1(NC(=O)NCc2ccc(C3(C(=O)OC)CCC3)cc2)CNCC12CCOCC2 c1(CC(C)C(N2CC3(NC(=O)Cc4csnn4)CCC2C3)=O)ccc(F)cc1F c1(-c2c(C)onc2)cccc2nc(C(=O)Nc3ccn4ncnc4c3)cn12 C(C1=NOC2(CCC2)C1)NC(C(C1CN(C(c2ccn(C)c2)=O)C1)O)=O CC#CCCCC(=O)N1CCCC(O)(CNC(C2(C)CC=CC2)=O)C1 C(=O)(CCCC(=O)C1CC1)NCCOCC(=O)NCc1c(C)nc(C)[nH]1 C(=O)(C(C)(C)CC(F)F)N1CC(C)C(C)(CNC(c2ccoc2)=O)C1 N1(C(CC)=O)CCC(NCc2csc(C)n2)CC1 CCC(C)(C)CC(=O)NC(c1ccccc1)c1nnc[nH]1 Cc1nn(C(F)F)c(C)c1C(=O)Nc1cnn(-c2ccccn2)c1C C(=O)(C1=C(Cl)CC1)NC(C1(NCc2nccn2-c2ccc(C(=O)O)cc2)CC1)C c1(C(N2CCCN(C(C3(CCOC)CC3)=O)CC2)=O)ccc(C)c(C)c1N Cn1cc2c(n1)CCC(C(=O)NCC(C1CC1)NC(=O)CNc1nccs1)C2 C(CC(COCc1ccccc1)N=c1nc(-c2cccc(C)c2)[nH]s1)OC c1(C(=O)NC(C(=O)Nc2ccc(OC)cc2)CO)ccc2c(c1)CC2 C=C1CCN(C(=O)C(C)=CCC)C(C(=O)NCC2=NOC(C)C2)C1 c1(C(=O)NCC(N(C)C(C2C=CCCC2)=O)C2CC2)cc(F)c(Br)c(Cl)c1 CCCC(CC)C(=O)NC1CC(F)CN(C(=O)CS(F)(F)(F)(F)F)C1 C1(NC(CCC(C)O)=O)CCN(C(C2CC=CCC2)=O)CCC1(F)F c1(C(=O)NC(C(C)NC(C=C(CCC)C)=O)(C)C)cc(OC)cc(Cl)c1F c1(COC)nnc2n1CCN(C(=O)C(=O)N(C1CSC1)C)C2 Cn1c(C(=O)N(CCOC2CN(C(=O)C(O)C(F)F)C2)C2CCC2)cc(Cl)c1Cl C1(NC(C2CCCCCC2)=O)CCC2(CCCNC2)C1 c1(C(=O)NCCNC(C(C(C)C)C#N)=O)cc2c(Cl)cccc2[nH]1 c1(C(=O)NC(C(C(C)C)NC(=O)COC2CC(F)(F)C2)C)ccc(O)c(F)c1 c1(CNC(C2CC3(CCCO3)C2)=O)ccc(CN2CCOCC2)c(F)c1 N1(C(C2(C#C)CCC2)=O)CCC(O)(CNC(C2CCC(F)(F)C2)=O)C1 C1(NC(CN(C)CC)=O)CN(C(=O)C(c2cscn2)N(C)C)CCC12CCC2 C1(CNC(C2CC2[N+](=O)[O-])=O)CCCC2CN(C(=O)CN3CCCCCC3)CC12 c1(CC(N2CCCC(C)(NC(C3CCCS3)=O)C2)=O)c(F)cc(F)cc1F c1(CC(=O)N(C2CCN(C(C34CC(OC)C3C4)=O)CC2)C)c(C)nc(O)nc1C c1(C(N2CC(CNC(c3ncc(Cl)nc3Cl)=O)(OC)C2)=O)c(F)cc(Cl)cc1F CCCCC(=O)C(=O)N1CCCC(NC(c2oc(CO)cc2C)=O)C1 N1(C(c2nc(C)c(C)[nH]2)=O)CC2CCC1C(CNC(=O)C(C1CC1)C1CC1)C2 C1(C2CCN(C(C3CC3Cl)=O)CC2)(NC(CCc2n(C)cnc2)=O)CC1 C1(C(=O)NC2CC(CNC(C(CC)OC)=O)C2)(OC(C)=O)CCCC1C c1(OC)cccc2c1OC(C(N1CC(CO)(NC(c3cncc(Cl)c3)=O)C1)=O)C2 N1(C(CCC(CC)NC(CCOCC)=O)=O)CCC12CCC(O)CC2 CC(C)(F)CCC(=O)NCC1(CNC(c2csc3nnsc23)=O)CC12CCC2 C=C(C)C1CCC(C)=CC1CC(=O)NCC(C12CCC(CC1)C2)NC(=O)CC Cc1cccc(N)c1C(=O)NC(C1CCN(C(=O)Cc2csc(Cl)n2)C1)C C1(CCC)CN(C(=O)C(=Cc2cccs2)C)CC1NC(c1c[nH]c(C)c1)=O CC(C)C(C)(O)C(=O)NC1CCCN(C)C1 C1(C(C)(C)CNC(=O)Cc2cocn2)CCN(C(c2cnnn2C2CC2)=O)CC1 C(C#Cc1cccnc1)NC(C1N(C(C(C(C)C)OCC)=O)CCC1)=O N1(Cc2c(OC)ccc(Cl)c2)CCCC2C(NC(=O)C=C(C)C)C(C)(C)C12 c1(C(=O)NC2CCN(C(C(C)c3cc[nH]n3)=O)C2)csc2ccc(Cl)cc12 N1(C(CCCc2cc(C)no2)=O)CCCN(C(=O)C(C)Cc2ccco2)C(C)C1 C(=O)(C1CCCc2ncnn21)N(C)CC1CN(C(=O)C=Cc2cc[nH]n2)CCO1 C1(C(=O)N(C)CC2(O)CCN(C(=O)C(c3cncn3C)O)C2)(OC)CCCCC1 c1(OC(C)C)ccccc1C(N1CCC(C)(NC(C2CCS2(=O)=O)=O)C1)=O N1(C(CNS(C)(=O)=O)=O)CCC(O)C(NC(=O)Cn2cccn2)C1 C1(C(N2CCC(=C)C2)=O)C2CC1N(C(=O)CCC1CCOC1)C2 C1(CC)CN(C(c2cc(C)cc(F)c2)=O)CCN1C(=O)Cc1ccsc1C C1(CNC(CCC(C)C)=O)COCCN(C(C23CCN(CC2)C3)=O)C1 C1(CCC)CN(C(=O)CN(C)C)CC1C(=O)NCCC1CCCC2CC12 C12(CNC(C(c3ccnn3C)NC(C(C)C#N)=O)=O)CCCC(CO1)C2 c1(C(N2CC(NC(CCCOC)=O)C(O)C2)=O)cnc2n1CC(C)CC2 Cc1cn2cc(C(=O)NCC3(C)CCCN(C(=O)CC4(O)CCOC4)C3)nc2s1 C(C(CC(C)C)NC(=O)C(C)n1cccn1)NC(c1ccc(CC(C)C)s1)=O CC1(NC(=O)C(F)CC2CN(C(C3NC(=O)OC3=O)=O)C2)CCOC1=O c1(OC)cc(C(N2CC(N(C)C(C3CCCS3)=O)C2)=O)nc(Br)c1 c1(CC(=O)NCC(CNC(CCC(=O)NCCC)=O)(C)O)cc(F)c(N)cc1F Cc1cc(-n2cc(COC3CCNC3)nn2)ccc1N C(CCCCCC(=O)NCc1cc(O)ccc1F)NC(c1cccc(C)c1N)=O C1(CC)CCCCCCN1C(=O)C(O)CCCNC(=O)CCC(C)C1CCC1 C1(C)(CNC(CN(CC)CC)=O)CN(C(=O)C(C(=O)OCC)(C2CC2)OC)CCO1 CS(=O)(=O)c1cccc(-c2cccnc2NCc2csc3ccccc23)c1 C1(C(=O)NCCCCN(CCCNC(CC(CC)SC)=O)C)CC(C(C)C)=NO1 C12(NC(C(C)Cc3ccco3)=O)CCC1CN(C(=O)Cc1ccc(Cl)c(F)c1)C2 c1(C(N(CCNC(C2CC(SC)C2)=O)C2CC2)=O)[nH]nc2c1CCCC2(C)C N1(C(COCc2nnc(C)s2)=O)C2CCC1CC(NC(C1(CO)CCCO1)=O)C2 CC(C(C)(C)C(=O)N1CCC(CF)C1)NC(=O)COCCF C1(NC(COCC)=O)CN(C(c2cnoc2C2CCOCC2)=O)CC2(CCC2)C1 C=C1CCC(CNC(=O)C(C2CCCCC2)NC(C2CC2C(=O)OCC)=O)CC1 C1(NC(C(CC)N(CC)CC)=O)(CO)CCN(C(C2(C(F)(F)F)CC2)=O)C1 C1(NC(CSCC(=O)NCCC(=O)OCC)=O)CCN(C(=O)C=CC)CC1 CCC(C)C(C)C(=O)N(CC(C)NC(=O)Cc1cc(C)[nH]n1)C N1(C(C(C)NS(CC)(=O)=O)=O)CC2(CCC(CNC(=O)CC3(C(F)F)CC3)O2)C1 C(CC(C)C)(C(=O)NCCOCCN(C(=O)CC(C)n1ccnc1CC)C)OC c1(C(=O)NCC(C)CNC(=O)CCc2nccn2C)coc(C#N)c1 C12(C(N(C)Cc3c(C)ncs3)=O)CCN(C(c3cn4c(n3)CCC4)=O)CCC1C2 C(C(=O)NCC1CCC1NC(c1[nH]c(C)cc1C)=O)(C(C)(C)C)OC C1(C(=O)NC2(C)CC(NC(C(C3CC3)OCC)=O)C2)(OC)CC(F)(F)C1 C1(OC(C)C(N2CCCC2CCNC(=O)CC23CCCC2C3)=O)CCCCC1 C(CC(C)(C)CN=c1[nH]c(=NC(C)c2cncn2C)[nH]c2cc(C)ccc12)OC c1(OC)cc(C(=O)NC2CCOCC2C(=O)N(C)Cc2ccncc2F)nn1C CCC(C)C(O)C(=O)N1CC(F)CC1CNC(=O)C(c1ccc(Br)s1)=O c1(C(=O)NCCCN(C(=O)CNC(c2nccn2C)=O)C)cncn1C.C(C)(C)(C)O CC1SCCC1NC(c1ccc(-c2ccco2)[nH]1)=O N1(C(C(C)CN2CCCCC2)=O)CCOCC(NCCc2cccc(I)c2)C1 C1(NC(c2c(C)csc2)=O)CN(C(c2ccoc2)=O)C2CC12 C1(NC(C(C)OCC=C)=O)C2COCC1CN(C(c1cc(C)ccn1)=O)C2 c1(C(N(C(C)CNC(c2cccc(OC)c2)=O)CC)=O)cc(C)n(C2CC2)n1 c1(C(N2CCCCC(NC(C(C)N3CCC3)=O)C2)=O)cc(F)c(F)cc1Cl CCCC(C(=O)OC)C(=O)N1CCCC1C1CCN(C(c2cnn(C)c2C)=O)C1 C(C1CCCN1C(C1CCCS1)=O)=CC(=O)N(CCC(C)(C)O)C c1(C(=O)NCC2CN(C(=O)C(F)(F)C3CCCCC3)C2)cnn2cnnc2c1 c1(C(N2CCC(CC(C)NC(c3n(CC)ccc3)=O)CC2)=O)cc(C)nc(C)c1 CC(=O)CCCCC(=O)N1CC(C(O)C(N2CCC(N(C)C)CC2)=O)C1 C1(CNC(C=CCC)=O)CC2(CCN(C(c3ccc(CN(C)C)o3)=O)CC2)CO1 N1(C(C(C)N(C)CC)=O)CCC2C1CCN2C(c1cccc(Br)c1F)=O C1(NC(C23CC(OC)C2C3)=O)CCC2(CCCN2C(=O)C(=O)NCC2CC2)CC1 c1(CNC2C(C(=O)Nc3ncc(C)nc3Br)C2)ccc([Si](C)(C)C)cc1 C(N=c1ccnc(C2CC2)[nH]1)C1CN(C(c2cn(C)c(=O)n2C)=O)CC12CCC2 N1(C(c2c(OCC)scc2)=O)CCC2(NC(=O)C3=CCSC3)CC2C1 C1(C(N2CC(N(C(C(C(C)C)NC(C)=O)=O)C)C2)=O)CCC2(CCC2)CC1 c1(CC)cccc(F)c1C(=O)NCC(CNC(C1(C(F)F)CCOCC1)=O)OC C12(NC(C3C(C)C(=O)C3)=O)COC(CNC(c3cnn(C4CCC4)c3)=O)(C1)C2 c1(C(=O)NCCC(C)NC(=O)CCc2ccn(C)n2)cnc2[nH]c(=N)sc2c1 N1(C(CCC)=O)CCOCC1C(N1CC(O)(CNC(=O)C=Cc2ncc[nH]2)C1)=O C#Cc1ccc(CC(N2CCCC2C2(NC(C3CCC=CCCC3)=O)CC2)=O)cc1 c1(C(=O)OC)ccc(S(=O)(=O)N2CC3CN(Cc4cccs4)C3C2)n1C CC1(C)CCCCC1=CC(=O)NC1(CNC(=O)CCN2CCC(F)C2)CCC1 c1(C(=O)NCC(CN(C(c2n(CC)ncc2Cl)=O)CC)(C)C)cc2occc2[nH]1 c1(OC)cc(C(=O)N(CCCCN(C)C(c2nccn2C(C)C)=O)C)cc(C)n1 c1(C(N2C(C(=O)NCc3cocn3)CCCC2)=O)cccc(O)c1O c1(N(C(=O)CCN(C)C(C23C=CC(CC2)C3)=O)CC)ccccc1C c1(N2CCC(n3c(C(N)=O)ccn3)CC2)ccnc(N2CCCCCC2)c1 C(CCCC(=O)N(C(C)(C(=O)N1CCC1(CO)CO)C1CC1)C)OCC CC(CCNC(=O)CC1CCN(C)CC1)CCNC(C1CC12CCC2)=O Cn1ncc(CNC(c2csc(Cl)c2)=O)c1C(=O)NCc1nccn1C1CC1 N1(C(c2ccc(O)cc2)=O)CCCCC1=CC(c1ccc(C)s1)=O N1(C(CC2ON=C(C)C2)=O)C2CCC1CN(C(=O)CC(F)(F)c1ccccc1)C2 C(CC(N)=O)(C(=O)NC1(CC)CCC1)NC(c1ncn(CC)c1)=O C(c1cn(C(C)C(=O)N(C)C)cn1)=CC(C(=O)Nc1ccc(SC)cc1)C c1(C(=O)NC(CC)(CNC(=O)Cc2sccc2C)CC)nccc2ccccc12 C1(NC(CCCCC)=O)CC2(C1)CC(NC(C1CCN(C(=O)C(N)=O)CC1)=O)C2 c1(C(=O)NC2CCC(CNC(C(C)n3cncn3)=O)C2)cc(O)ccc1[N+](=O)[O-] c1(C(N(CC(C)C)CC(=O)N(CCO)N)=O)ccnn1C.C1CC1 C1(NC(c2cnc(C3CCOC3)s2)=O)CN(C(c2cncc(Cl)c2)=O)CCC1F CCCC(C(=O)NC(C1(CC)CC1)C)OCC.C12(CC1)C(=O)N2.OCC Cc1nc2cc(C(N3C(CNC(=O)CNC(N)=O)CC4CC34)=O)ccc2o1 O=C1CC(C(=O)NC2CC(O)CN(C(C3CC(=O)N(C4CC4)C3)=O)C2)=NN1 C1(CC)CN(C(=O)C=CS(=O)(=O)CC)CCC1NC(=O)C(C)(C)C(F)(F)F C1(NC(C(N)=O)=O)COC2(CCN(C(=O)CCN3CCCCC3=O)CC2)C1 c1(C(=O)NCC(N2CCN(C(C(CCC)O)=O)CC2)C)ccc2n[nH]cc2n1 C12(C(N3CC(C)C(NC(C4CCSCC4)=O)C3)=O)CC(C)(C1)OC2(C)C c1(C(CNC(C2CC2F)=O)NC(CC(C)NC(C)=O)=O)ccc(C(C)C)cc1 c1(OC)cc(CNC(c2cc(Cl)ccc2Cl)C)ccc1OCc1ccccn1 CCCC(F)C(=O)NC(Cc1ccco1)C(=O)NCC1CCC(=O)N1 C1(c2cnn(C)c2)(CNCCC#CC)CCCO1 CON1CCC(CC(N2CCC(O)(CCNC(c3nc(C)nn3C)=O)C2)=O)CC1 C(CC(C)N=c1[nH]c(C)c(C(=O)O)s1)NC1CCC(C)C1 CC1CCC(CNC(=O)COCc2cccnc2)N(C(c2cncc(O)c2)=O)C1 C(=O)(C#CC(C)(C)C)NCCOCc1cn(C2CN(C(C(CC#C)C)=O)C2)nn1 c1(C(=O)NCc2ccc(C)cc2Cl)nccc2c1NCCC2 c1(C(=O)N(CC2C3CN(CCN4CCCC4)CC23)CC2CC2)ccc(F)c(Cl)c1 c1(C(N2CCCC(NC(CCCOC(C)=O)=O)CC2)=O)coc2c(Cl)cccc12 C(=O)(C(C)(C)C(C)(F)F)NCC1N(C)CCN(C(c2ccc(O)c(CO)c2)=O)C1 C1(CNC(C2C(C=C)OCC2)=O)(NC(=O)CC2CN(C)C2)CCCCCC1 N1(C(C2C(NC(CCc3nc(=N)[nH][nH]3)=O)COCC2)=O)CCC(CO)C12CC2 C1(C(=O)NCC(N(C)C(c2n[nH]cc2Br)=O)C2CC2)CC2CC(=O)C1O2 C(=O)(C#CC1CCCOC1)N1CCN(C(c2ccc(F)cc2F)=O)CC1CCO N#Cc1cscc1C(=O)NCC1(CNC(C2(O)CCSC2)=O)CC1 O=C(C1CSc2ccccc21)NC1CC2CN(C(C3CCCC34CC4)=O)CC12 C1(CC#C)(C(N2CCCC2CN(C)C(C23CCN(CC2)C3)=O)=O)CCOCC1 Cc1ccc(F)c(O)c1C(=O)NCCN(C(=O)CCc1cccnc1C)C(C)C C1(C(=O)NCC2(CN(C)C(C3CC(F)(F)C3)=O)CC2)CCN(c2ccncc2)C1 c1(C(N(CC=CC(=O)O)C)=O)ccc(C(=O)O)c(Cl)c1.N1(CC(C)=C)CCOCC1 c1(C(=O)NC2C(NC(COCC#C)=O)COCC2)cc(OC)c(OC)c(Cl)c1 C1(NC(C2C(OCC)CC2)=O)CN(C(c2cnncc2O)=O)C(CC)(CC)C1 C1(C(C(=O)N(CCCCCNC(C2(O)COC2)=O)C)F)CCCCCC1 C1(NC(c2c(COC)cco2)=O)CCCCN(C(c2cc(OC)n[nH]2)=O)C1 C1(C(=O)NC(c2ccncc2)C)CN(C(=O)C(c2ccco2)SC)CCC1(C)C N1(CCC)CCCC(C(=O)NCCOCCNC(=O)C#CC(C)C)C1 c1(OCC(=O)OC)ccc(NC(=O)C(CC(N)=O)c2ccccc2)cc1[N+](=O)[O-] c1(CC(=O)NC2CN(C(c3c(CC)c[nH]n3)=O)CC2CC)cncc(C#N)c1 N1(CC(=O)NCC(F)F)CCCC1c1ccsc1 C(C(=O)NC1CCC(F)(F)CC1)(C1=NOC2(CCC2)C1)N1CCC(C)(N(C)C)C1 C1(CNC(c2c(OC)cc(C)s2)=O)CN(C(c2cnc(C)[nH]2)=O)CCCO1 N(C1CCOc2c(F)cccc21)C(N(CC(C)OC(C)(C)C)C)=O c1(C(=O)NC(CN(C(=O)C(c2cncn2C)O)CC)C)cccc2sccc12 N1(S(C(C)C)(=O)=O)CCCCC1C1CCCN(C(C2CCC2(F)F)=O)C1 c1(NC(CC(C)NC(C2COC(C)(C)C2)=O)=O)ccc2c(c1)CCC2 C#Cc1cccc(CN(C2CCCCC2C)c2ccc(F)cc2)n1 c1(C(N(C(CN(C(c2cc(CCC)on2)=O)C)C)C)=O)ccc(N(C)C)nc1 n1(CC(N(CCNC(c2ccc(C#N)cn2)=O)CC)=O)nc2n(c1=O)CCOC2 C1(COC)(NC(=O)CCCC(=O)NCC(C)C)Cc2ccccc2C1 Cc1ccc(C(=O)NC2CCN(C(=O)CN=S(C)(C)=O)CC2C)c2c1CCCN2 S(=O)(=O)(c1cnccc1NC1CCCc2cnccc21)N1C(C)SC(C)SC1C c1(C(=O)NCC(=O)NC(C2CCN(C(=O)Cc3ncnn3C)C2)C)ccncc1 c1(C(N2CC3CC4C(NC(CC5(C)CC5)=O)C2C3C4)=O)ccc(Cl)c([N+](=O)[O-])c1 N1(C(CSc2cn(C)nc2)=O)CCC(NC(=O)C(C)(C)C2CCCO2)CC(O)C1 N1(C(c2cc(CC)ncc2)=O)CCOCC(C(=O)N(C)C(C)C2CC2)C1 c1(OC)ccc(F)c(C(=O)NCC2CCCCC2NC(C23CCC2CC3)=O)c1F C1(C(=O)NCc2c(C)nsc2)CCCCN(C(c2coc(COC(C)C)n2)=O)C1 Cc1nc(C(=O)NC2CN(CCCC3CC3)CC2O)ccc1Br c1(CC(=O)NC(CC(C)C)CNC(=O)CN2CCCC2=O)cccc([N+](=O)[O-])c1 N1(C(c2c(C)ncnc2)C(=O)NCC2CC2)CCCC(Cc2ccccc2)C1C CC(C)CC(C)(O)C(=O)NC1(C)CN(C(=O)C(F)(F)C2(O)CCC2)C1 c1(C(N(C(C)CNC(=O)C(Cc2ccccc2)OC)CC)=O)ccc(N)cc1Cl N1(C(c2cc(OC)c(OC)cc2)=O)CCCC(NC(C2C=CCC2)=O)CCC1 c1(C(=O)NC2C(C(=O)NC(CCC)C3CCC3)CC2)cnc(C)nc1C C(C)(C(=O)NC(c1nccs1)C)(N(C(C(C)c1cc[nH]n1)=O)C)C1CC1 Cc1cc(C)c2cc(N3CCC(c4nc(-c5ccc(Br)cn5)no4)C3)[nH]c2c1 C1(NC(c2cn(C)nc2)=O)C2CC3C(C2)C13C(=O)NCC1CC12CC2(F)F C1(CNC(CC2(C)CC2)=O)CCC(F)(CNC(c2ccc(Cl)nc2)=O)C1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(=O)Cc1csc(S)n1 N1(C(c2cc(CCN(C(CCC(N)=O)=O)C3CC3)on2)=O)CCC(F)(CF)CC1 C(=O)(C(C)C1CCC1)NCC(=CC(=O)NCC1(CCOC)CC1)C N1(C(C(CCOC)C)=O)CCC(NC(=O)CSCCOC)CC1C C1(CNC(C2OCCN(CC)C2)=O)CN(C(=O)C(C)=O)CCN1C C1(N(CC#C)C(c2cnc[nH]2)=O)CCN(C(C2CC(CN(C)C)CO2)=O)CC1 c1(CC(=O)NCC(=O)NCCn2cc(-c3ccccc3F)nn2)ccc(Cl)c(Cl)c1 C(=O)(C1=COCCO1)NCCc1c(CNC(C2(OC)CCCC2)=O)nco1 C1(C(N2CCN(C(c3cnsn3)=O)C3CCCC23)=O)CCc2cc(F)ccc2O1 C(=O)(C1=CC2(CN(C(c3ccn4ccccc34)=O)C2)OC1)NCC(C=C)O C1(NC(C(C=C)(C)C)=O)CC(C)CN(C(c2ccc(C(=O)OC)c(F)c2)=O)C1 Cc1cnn(C)c1CC(=O)NC1CCOC(CNC(c2cc(C(C)C)no2)=O)C1 Cc1nn(CC(=O)NCc2cc(C(=O)NC(C3CCCC3)CO)n(C)n2)c(=O)o1 C1(NC(CCCSC)=O)CC2CCC(C1C)N2C(C1CCN(C(N)=O)CC1)=O C1(N(C(CC(CC)C)=O)C)CN(C(C2(F)CCC2)=O)CC1(C)C N1(C(c2cn(C)nn2)=O)CCc2sc(CNC(C3CC4(C3)CC43CC3)=O)nc2C1 c1(OC)ccc(Cl)cc1C(=O)NC1CC2CCC1N2C(=O)CC1CCC(=O)N1 c1(C(=O)NCCCN(C(c2cnc(C(C)O)s2)=O)C2CC2)cc2c(ncn2C)[nH]1 C(=O)(NNc1ccc(NC(=O)OC(C)(C)C)cc1)C1(CO)C(OC)CCCCC1 CC1(NC(=O)CCSc2ccc(Cl)cc2)CCN(C(=O)CC2(C)CC2(F)F)C1 N1(C(c2c(NC)nccc2)=O)CCC2(CC1)CC(NC(C)=O)C2 N1(C(C(CN(C)C)NC(CCCC#C)=O)=O)CCC2(CCOC2=O)C1 N1(C(C2CCN(C)C2)=O)CC(NC(=O)CC2CN3CCC2CC3)CC2(CC2)C1 C1(N(C(c2cnn(CC(F)F)n2)=O)CC)CCN(C(=O)Cn2cc(CO)nn2)C1 C1(NC(c2cc(CC)n(C)n2)=O)CC2CC1N(C(c1sc(OC)nc1Cl)=O)C2 C1(N(C(C=Cc2c(C)ccs2)=O)C)CN(C(c2sccc2C(C)C)=O)CC12CC2 N1(C(Cc2cn(CC)nc2)=O)CCCC(CC)C1C(=O)NCC(C)N(C)C C1(NC(CC2N(C)C(=O)CC2)=O)CCC2CN(C(=O)C3=COCC3)CCC2C1 Cc1ccc(CCC(=O)NC(C)CCN(C)C(C2(Br)CC2(F)F)=O)cc1 N1(C(C(=O)NCCC)C2CC2(C)Br)CCc2c(ccn(C)c2=O)C1 C1(C(N(C2CN(C(=O)Cc3cccc(OC)c3)C2)CC)=O)COC2COCC12 c1(C(=O)OC)nc2ccccc2nc1N(C)Cc1c(F)cccc1F C1(NC(C=CC(C)(C)C)=O)(NC(=O)CNC(=O)NCc2ccco2)CCOC1 Cc1nn2cc(CC(=O)Nc3cccc(NC(c4csc(Cl)n4)=O)c3)nc2s1 CC(Cc1cccs1)C(c1nnnn1Cc1nnn(C)n1)NCCC(F)F c1(NC(c2c(C)nccn2)C)[nH]c(=NCc2nnc(CO)s2)nc2scnc12 NS(=O)(=O)c1cc(C(=O)NCC2CCCCN2C(C2CC2(F)F)=O)c(Cl)o1 C1(NC(c2ccc(N(C)C)nc2)=O)CC2CC(C1)N(C(=O)Cc1nccn1C)C2 c1(NC(C)=O)ccccc1CNCc1nc(-c2ccccc2)oc1C c1(CC)ccc(C(=O)NC2CCC(C(N3CCC(CC(C)(C)C)C3)=O)CC2)c(Cl)n1 C12(CNC(C(C)(C)c3ccccn3)=O)CC(CN1C(c1ccc[nH]1)=O)C2 C1(CC(=O)NCCN(CCOCCO)C(c2ncc[nH]c2=O)=O)CCCC(F)(F)C1 N1(C(C2CC(OC)C2)=O)CCC2(NC(=O)Cc3ccns3)CC2C1 C1(C(=O)Nc2cnn(C(C)C)c2C)(CC)CCCN(C(c2cncc(O)c2)=O)C1 c1(C(N2CCN(CCCNC(C3CC3C3CC3)=O)CC2)=O)ccc2c(c1)CC2 c1(NC(C2CCCCN2C(=O)Cc2ccc(F)cc2)C)ncnc2c(Br)cccc12 CCC(CC)C(C)C(=O)NC(C)CNC(=O)C(O)(C(F)(F)F)C1CC1 C1(N(C(C(C)OCCC=C)=O)C)CCCN(C(=O)CCN2CCCC2=O)C1 C(CC(=O)NCCCCN(CCCNC(C1(NC(N)=O)CC1)=O)C)SC S(=O)(=O)(c1cnn2ccc(=NCCN3CCCS3(=O)=O)[nH]c12)NCCSCC Cc1cc(O)c(Cl)cc1C(=O)NC(CNC(c1c[nH]nc1C)=O)C(C)C(C)C N1(C(=O)NC2C(c3onc(CC)n3)C2)CCNCC1C1CCOC1 CC1(C)CC2(CO1)CN(C(=O)NCC1CCOCC1F)C2 O=C(C#CC1CC1)NCc1ocnc1C(=O)NC1CC1CO Cn1cc(CC)cn1.c12c[nH]c(c1)C(=O)NCC(=O)NC(C)(C)CNC(=O)CC2 C1(CC)CN(C(c2ccc3nsnc3c2)C(=O)Nc2ccccc2)C2(CCC2)C1 CN1CC=CCC1CC(N1CCC(NC(c2ccc(CO)s2)=O)C1)=O c1(C(N(CCCNC(=O)C(O)CF)CC)=O)cccc(-c2ccccc2)c1F C1(CNC(CSCC#C)=O)CC2COCC2N1c1cc(COC)nc(C)n1 c1(C(N2C(CNC(C(c3n(C)ncc3)O)=O)CCC2)=O)ccn2c(O)nnc2c1 N1(C(C=C(C)Cl)=O)CC2CCCC2(NC(=O)Cc2cc(F)c(F)c(F)c2)C1 C1(NC(=O)CCc2ccncn2)C2CCN(C(=O)C3CC3)CCC12 C1(CC)CN(C(c2cnc[nH]2)=O)CCN1C(C)=O c1(C(N2CC(CC(=O)NCCc3cccc(O)c3)C2)=O)cc2cc[nH]c(=O)c2s1 N1(C(C(CC=C)NC(=O)C(F)=CC2CC2)=O)CC2NC(=O)OC2C1 C#Cc1ccc(C(=O)NC(CNC(=O)C(O)C(C)(C)C)CC)c(C)c1 c1(OC)cnc2ccc(C(=O)NCCC(C)N(C)C(c3coc(Cl)c3)=O)cc2n1 N1(CCC(=O)NCC(F)CNC(C2CC3CC3C2)=O)C(=O)CCC1=O C1(C(=O)NCC(CC(=O)OC)C)CC(O)CCN1C(C1CN(C)C1)=O C(=O)(C1=NNC(=O)CC1)N1CCC(CNC(c2c(CCC)n[nH]c2)=O)(COC)C1 C(=O)(C(C)(CNC(C1CNC(=O)C1)=O)CC)NCCCOCCCC c1(NC(C(C)C)CC(F)(F)F)ccc(S(=O)(=O)N2CCCCC2CF)cc1C#N C1(CNC(c2c(C)con2)=O)CC2CCC1N2C(C1COC(=O)O1)=O N1(C(=O)CSCc2cscn2)CC2CCC(C1)N(C(=O)CO)C2 c1(C(=O)NCCOc2ncccn2)cccc(NC2CS(=O)C2)c1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(NC(C2CCCC2C)=O)C(O)C1 C(CCC1CC1)(C(=O)NCC1(O)CCCOC1)NC(COCCCCC)=O N1(c2nc(OCC)c(Br)cn2)CCCC(C2CN(C(=O)CCc3cnc[nH]3)C2)C1 n1(CC)cc(C(=O)NCC(CO)NC(c2cc(C(C)C)oc2C)=O)c(C)n1 C12(C(=O)NC3CC(CNC(C(C)(C)OCC)=O)C3)CCCCC1C2(F)F CCC(C(=O)NCc1nc(C2CCN(C(c3cccs3)=O)CC2)n[nH]1)CO C(=O)(C1=NNC(=O)CC1)NC(C1CCCN(C(C2(COC)CC2)=O)C1)C N1(C(CC=C=C)=O)CCCC2(CCN(C(=O)Cn3cc(S(C)(=O)=O)cn3)C2)C1 Cc1cc(C(=O)NC2(C(=O)NCCC(=O)OC(C)(C)C)CCCC2C)cnc1C c1(C(C(=O)OC)NC2(CO)CCC2)cccnc1 C(=O)(CCCC(F)(F)F)N1CCC(CNC(c2cc(F)c(Br)cc2F)=O)C1 C12(C(C)(C)C1(C)C)C(=O)NC2.C1(C(=O)OCC)(OC)CC1(F)F c1(OCC(=O)NCC2N(C(C(COC)OC)=O)CC=C2)c(Cl)cc(Cl)cc1Cl C#CCC(C(=O)NC(C)CS(N)(=O)=O)NC(=O)Cn1cncn1 c1(CC)nc(C)c(C(=O)NC2CCC(CNC(c3ccc(C(C)C)cc3)=O)C2)o1 N1(CC(=O)NC(C2CCCC2)CNC(C(C)CF)=O)C(=O)CCC1=O O(NC(=O)C(CCN(C)C)NC(=O)C(=CC1CCCC1)C)CCC#C C1(C(C)C)C(C(=O)NCC(C)(C)C2CCC2)CCN1C(C1CN(C2COC2)C1)=O c1(C(C(=O)NCCC#N)N(CC(F)Cl)C)cn(C)nc1Br C=Cn1ncc(C(=O)NC2(C(=O)NC3(CCF)CC3)CC2C)c1N C(=O)(C1=CC2(CCN(C(c3cc(O)ccc3C)=O)C2)C1)NCC(C#C)C(C)C c1(SCCN(C(=O)CSc2ccncc2)C)ccc(Cl)c(Cl)c1 c1(OC)cccc2c(C(=O)NCC(C)(Cc3cccs3)CO)csc12 N1(CCCCNC(=O)CC2CCCOC2)CCCN(C(c2ccccn2)=O)CC1 CCCCCC(=O)NCC(N1CCCC1C1CCN(C(=O)CC(C)SCC)C1)=O C1(C(N(CCNC(c2ccn(C(F)(F)F)n2)=O)C2CC2)=O)OC2CCC1C2 c1(C(N2CCCC(F)(C(=O)NCC3(C)CCCO3)C2)=O)cncc2[nH]ccc12 N1(C(CC=CC=C)=O)CCC(CCC2CCN(C(=O)C(C)C(C)C)CC2)CC1 C1(C(N2CCC(O)(C(C)NC(=O)CC3CCS(=O)(=O)C3)C2)=O)C2CC3C(C2=O)C13 C(=O)(CCCC(=O)NCC1CCCN1C(=O)CCc1cc(C)no1)NCC N1(C(C(C)OCCCC)=O)CCCC(NC(=O)CCc2ccn(C)n2)CCC1 N1(C(c2ccccc2-c2ccc(Cl)c(F)c2)=O)CCc2c(F)cc(Br)cc2C1 CC(C(C)(C)c1cccs1)NC(=O)CC1CCC(C(=O)O)C1 C1(CN(C2CCCCC2)CC=C)CC2(C1)CC(C(F)(F)F)C2 C1(CN(C(=O)NCC2CCC(C)CO2)C)CC12CCOCC2 CCC(C)C(C(=O)N(CCCCN(C(=O)C#CC(C)(C)O)C)C)N(C)C.C1CN1 c1(C(=O)NC(C2CCCC2)CNC(C(C2CC2)OC)=O)c[nH]c2c(C)cccc12 N1(CC(N2CC3C(N(C(=O)CCCS(N)(=O)=O)C)C3C2)=O)CCCC2(CC2)S1(=O)=O C(=O)(C(CC)C(C)(C)CC)N1C(CCC)CN(C(c2cncn2C(C)C)=O)CC1 CC(CO)(CO)C(=O)N1C2CCC(C2)C1C(N1CCOC(CO)C1)=O C(=O)(C1CCCn2cncc21)N1C(C)CC(CNC(c2c(C)cnnc2)=O)C1 N1(C(=O)C=Cc2cccs2)CC2CCC1C1CN(c3ncncc3Br)CC21 C1(CC)CN(C)CCN1C(C1CCC1NC(C1CC12CC2)=O)=O CCCC(CCC)CCCC(=O)N(CC(O)CNC(c1ccnc(F)c1N)=O)C c1(C(=O)NC2C(NC(C(C)(C3CC3)OC)=O)CCC2)nc(Br)c2ccccn12 c1(C(=O)NC2(C)CCCN(C(c3ccn(C)c(=O)c3)=O)C2)ccc2[nH]ccc2n1 C1(C)(C(=O)NCCCCN(C)C)CCN(C(c2c(F)cncc2Br)=O)CC1 Cc1nccc(C)c1NC(C1CCN(C(=O)C(C)Cn2cccn2)C1)=O CC(CCNC(C1CCCN(C(c2n[nH]c(O)n2)=O)C1)=O)C(F)(F)F C1(C(=O)NC2CC3CC(NC(CCC4CC(C)C4)=O)CC32)CC2CCC1C21CC1 c1(CC)cc(C(=O)NC2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)C2)ncn1 c1(C(=O)Nc2ccc(CC)cn2)cccc2[nH]nc(-c3c(CO)cccc3F)c12 C(N=c1[nH]c(=NCCC2CCCC2)[nH]c2ccsc12)c1cnc(CC)[nH]1 C(=O)(C(C)(C(C)C)OC)NC1C(NC(COC)=O)CCC1.C1(C)CC(SC)C1 c1(N(CCCCF)C)ncnc2c1ncn2C1CC(O)(C(F)(F)F)C1 C1(C(=O)NC(c2ccns2)C)COCCN(C(c2nc[nH]n2)=O)C1 Cc1c(C(N2C(C(=O)Nc3cnn(C)c3C(C)C)CC2C)=O)cccc1F C1(C(N2CCC(N(C(c3cccc[n+]3[O-])=O)CC)C2)=O)CCC2(CCC2)C1 N1(C(Cc2nc(COC)sc2)=O)CC(NC(c2ncccc2C)=O)C2CC12 N1(C(CCOC(CC(C)C)C)=O)C2CCC1CN(C(=O)CCC(F)F)CC2 O(C=CC(=O)NCC1CCN(C(C2CCC2C(F)F)=O)C1)CC CC(C(=O)N1CC=CC1C(=O)NCC(=O)N1CCCO1)C(F)(F)F C=Cc1ccc(C(=O)NCC2(C)CC(NC(C3CCOC3(C)C)=O)C2)cc1 CC(C)(C)C(C(=O)N1CC2C(C1)C2(F)F)NC(=O)C=CC(=O)NC1CC1 CCS(=O)CC(=O)NC(c1ccc(Cl)n1C)c1nnnn1CC(F)F c1(SCC#N)ccsc1C(N1CCC(NC(=O)CN2CCCC2CO)C1)=O n1(CCC)cc(C(=O)NC2CCC2NC(c2cn(C3CCN(C)C3)nn2)=O)nn1 C(=O)(C1CCc2cccc(O)c21)NC1CC(NC(c2cc(C)nn2C2CC2)=O)C1 CCCN=C(NCC(c1ccccn1)C)N1CCCC(O)(CO)C1 C(Cc1csc(Br)c1)(C(=O)N1CCOCC1)N(C)CC1CCCN1C1CC1 c1(OC)ccc(N(CCO)C(=O)NCCC(O)CO)cc1SC C(=O)(CCC(C(C)C)NC(=O)CCP(C)(C)=O)NCc1n[nH]c(C)c1C C1(C(N(CCC2N(C(C(C)NC=O)=O)CCCC2)C)=O)CCC2(CC1)CC2 N1(C(COCC(=O)OC)=O)CCOCC1CNC(=O)CCC1CC1(C)C CCC(CC)C(C)C(=O)NCC1CCN(C(=O)CC2CCOC2C)C12CC2 C123CCCC(CN1C2)C3.c1(OC)cc(C)nc(Nc2cc(C)nn2C(C)(C)C)n1 c1(C(C(=O)NCC(C2CCCC2)NC(C2C(OC)C2)=O)C)ccccc1C S(=O)(=O)(c1cnc(NCCN(C)CCO)c(Cl)c1)N1CC(CC)SCC1 Cn1cnc2cncc(C(=O)NCc3cccc(CNC(C4CC(F)C4)=O)c3)c12 c1(C(=O)NC(CC)CN(C(=O)CCCCC(C)(C)C)C)cc2cc(C)ccc2o1 C1(N(CCS(=O)(=O)N(C)C)CCO)CCC(n2cc(C3CCCC3O)nn2)CC1 N1(C(CC(CC)C)=O)CCC2(CC2NC(C2CC23CCSCC3)=O)C1 Cc1c(C(=O)NCC2C3CN(C(=O)C(C)(C)F)CC23)nc(O)c2ccccc12 c1(C(=O)NC2CN(C(c3sc(C)c(O)n3)=O)CC(O)C2)cnc2sccn2c1=O C=CC1CCCCN1C(=O)C(F)CC1N=C2C(=CNN2)C(=O)N(C)C1 C1(CC)(NC(=O)Cn2ccnn2)CCCN(C(C2CC2c2ccncc2F)=O)C1 C1(C(=O)NCC2(CNC(c3c(C(C)C)ocn3)=O)CCC2)CCc2c[nH]nc2C1 c1(N2CC(C)N(CCOC)C(C)C2)ncnc2cc(Br)cnc12 C1(C)(NC(c2cc(-c3cn(C)nn3)on2)=O)CCN(C(C2CCC(=O)C2)=O)CC1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2ncn(C(C)C)n2)=O)ncc1F N1(C(c2c(OC)nc(Cl)cc2)=O)CC2CCN(C(=O)Cc3csc(S)n3)CCC2C1 CC(C)C(C(=O)NCCN(C1CCCC1)C(C1CCCN1C=O)=O)n1cncn1 N1(C(c2c(C)cc(F)cn2)=O)CC2CCOC2(CNC(=O)CC2CCOC2)C1 c1(-c2n(CC)ncc2)ccc2ccn(CC(=O)Nc3ccc4[nH]nc(Br)c4c3)c2c1 C12CCN(C1)C(=O)C(=O)N2.c1(CC(C)Sc2cccnc2)nncn1C N1(C(c2cnc(C)s2)=O)CC2C(NC(=O)CC(C)CC(C)C)CS(=O)(=O)C2C1 CCC(C)C(O)CC(=O)NCC(C)(C)CC(=O)N1CCCC(CC)C1 CC1(C2CCN(C(=O)CC3CC3Cc3nn[nH]n3)CC2)COC(=O)N1 CCC(C(=O)N1CCC(CN(C)C(c2cc(-c3ccoc3)[nH]n2)=O)C1)OC c1(OC)ccc(C(=O)NC(C2CN(C(=O)CC(C)CF)C2)C)cc1O Cc1cc(N)cnc1C(=O)N(CC(C)NC(c1sc(C(F)(F)F)nc1C)=O)C c1(CC(=O)NCC2(C)CC(NC(c3cn(CCC)nc3)=O)C2)c(Cl)cccc1Cl c1(NC(c2c(C)onc2)=O)cccc(-c2ccc(-c3ccccc3)o2)c1F C(=O)(C(C)(F)C(F)(F)F)NCCC1(OC)CN(C(c2scc3c2OCCO3)=O)C1 c1(C(CF)NC(=O)CC2CCCC2C(F)(F)F)ccccc1 c1(OC)cc(NC(c2ccc(NC(c3cc(Cl)cc(I)c3)=O)nc2)=O)cc(O)c1 CCC(C(C)(F)F)NC(C1(C)CCN(C(C2CC(OC)C2)=O)C1)=O C1(NC(c2ccc(CCCC)cc2)=O)CN(C(=O)C(O)CSC)CC1(C)C Cc1ccnc(C(=O)N(C)CC2CCCN(C(c3nc(C(C)C)oc3C)=O)C2)n1 C(=O)(C1CC(O)c2ccccc21)NCC1(CC)CN(C(=O)C(CCOC)OC)C1 c1(OC)ccc(N(C)C)cc1.N12CCSCC1CCCNC(=O)C2 c1(CCOCCCO)ccc(C(F)(F)F)cc1.C1(CO)CN1 O=NN1CCCCC1C(N1C2CCC1C(CNC(C1CCCCC1)=O)C2)=O CC1CCCN(C(=O)C(C)N(C(=O)C(c2ccccc2)C)CC2CC2)CC1 C(C(CNC(=O)C(C1CCCCC1)O)CO)NC(C(C)=CC)=O C#Cc1ccc(Cl)c(C(=O)NCC2(F)CCN(C(=O)CCN3CCC3)C2)c1 c1(C(=O)NC(C2N(C(C3CC(C)OC3)=O)CCC2)(C)C)nc(C2CC2)ncc1Cl C1(C(N(C2CCN(C(=O)Cc3cccc(Br)c3)CC2)C)=O)CC12CCOC2 C#CC1CN(C(c2cc(C)nn2CC)=O)CCN1C(C12CCCCC1C2)=O c1(C(=O)NC2CCC(n3cc(-c4cc(C)sc4)nn3)C2)cc(Cl)cc(Br)c1 CC1=C(C(=O)NCC2CC3(CC(NC(C4(C)CC(C)C4)=O)C3)C2)CCCO1 CCC(CC)CCCC(=O)NC(c1cnn(C)c1)C(N1CCOC(CCO)C1)=O NS(=O)(=O)CCCCCNC(=O)C(=O)Nc1c[nH]ccc1=O C(=O)(CCCC(C)=O)NCC1C(CNC(CC2N(CC)CCOC2)=O)C1 N1(CC(c2cscc2F)=O)CCOC2CCCCC12 c1(C(c2cn(Cc3nnc(C)s3)nn2)N(C)C)ccnc2[nH]cnc12 C(=O)(C#CC1CCCCO1)N1CCC(C)(NC(=O)COc2ccsc2)C1 c1(C(=O)OC)[nH]c(C)c(C(=O)CN(CCc2ccc(Br)cc2)CCN(C)C)c1C C1(C(=O)Nc2ccc(C(N)=O)nc2)CC2CCC(C1)N2C(=O)CCc1cnoc1 C(N=c1[nH]c2cccc(Br)c2o1)C1C(NC(C2C(=C)CC2)=O)CCCC1 c1(C(=O)NCC2(F)CC(CNC(C3(C(=O)OCC)CC3)=O)C2)ccc(C)cc1Cl O=c1cc(CN2CCn3cc(C4CC4)nc3C2)nc2ccc3c(n12)CCCO3 CC(C)C1=NOC(C(=O)N(C2CC2)Cc2cn(C(c3csnn3)C)nn2)C1 C1(C(=O)NC(C)(CNC(c2csc(C#N)c2)=O)C2CC2)C2(CCC2)C12CCC2 C1(C(=O)NC2CN(C(CC(C)OC)=O)C2)COC2COCC12 Cc1ccc(C)c(CN(C(=O)CC2CC=CC2)C)c1.N12CCCC(C1)C2=O N1(C(C2(CC)CC(C)(C)C2)=O)CC2(C1)CN(C(=O)COCC1CCC1)CC2CO N1(C(CC=C=C)=O)CC2CN(C(c3nnsc3-c3ccccc3)=O)CC2(C)C1 CC(C)(CCC(=O)NC1CC(NC(C2CCC(=O)C2)=O)C1)[N+](=O)[O-] O=C1CCC(C(=O)NC2C3CCC2N(C(c2nc(C4CC4)ncc2Cl)=O)C3)=NN1 CC1(C)CCN(C(C2CCSCC2)=O)C1C(N1CC(N2CCCC2=O)C1)=O C1(C(=O)NC2C(C)(CC)C2)CCN(C(=O)CC2CCCN(C)C2)CC1C N1(C(c2n(CC)cnn2)=O)CC2CCC1C(CNC(c1cnc(O)n1C)=O)C2 CCCCCCC(C)CC(=O)NC(C)CNC(=O)C1=CCN(C)C1 N1(C(Cc2c(C)nccc2)=O)CCN(C(c2ccnn2C)=O)CC(O)C1 CC1(C)CCC(F)(F)CC1NC(c1ccc2c(c1)NCC2)=O c12ncccc1N2.c1(CN(CC(=O)N(CCC)C)C)nc(-c2cccs2)oc1C C(c1ccsc1)=CC(=O)NC(C)C c1(C(N2C3C(CNC(C(C4CC4)OCC)=O)C(C3)C2)=O)cc(Cl)cc(Cl)c1N C(=O)(CCC(=O)NC1CCN(C(=O)CCN2CCN(C)CC2)C1)OCC CC(C1CCCCC1)=CC(=O)NCC(F)CNC(=O)C(=O)NC1CCOCC1 N1(C(C(C)OCc2ccccc2)=O)CCCCC(NC(c2cc[nH]n2)=O)C1 C1(CNC(c2c(C)nsc2)=O)CCCN(C(C2(C(F)(F)F)CC(O)C2)=O)C1 c1(CCSC)ccc(F)cc1C(=O)SC1(CCO)CCCCC1 C(CC(C)C(=O)NC(CNC(C1C(C(=O)NCC)C1COC)=O)CC)=CC c1(C(=O)NCCN(C(C2(c3oncc3C)CC2)=O)CC)ccnc2ccccc12 c1(C(c2ccccc2)NC(=O)Nc2cncc(C(F)(F)F)n2)cc(Cl)sc1Cl c1(C(=O)NC2C(NC(CC=C)=O)COC2)cccc(C#CCO)c1 C=CCCCC(=O)NNc1cccc(C)c1C.O([Si](C)(C)C(C)(C)C)C(C)CNCC N1(C(CC=C)=O)CC2CCC(CNC(=O)C=Cc3ccnn3C)(C2)C1 C1(C(N2CCCC(N(C(=O)Cn3ncnn3)C)CC2)=O)CC2CC1C1CC21 C1(N(C(Cc2cnc(C)s2)=O)C(C)CO)CC2CNC1C2 CN1CC(C)(C(N2CCCC(Cn3cc(-c4cccs4)nn3)C2)=O)CCC1=O c1(C(N2CC(CN(C(CCOCCOC)=O)C)OCC2)=O)c(F)ccc(F)c1Cl c1(NC(C(=O)NC(C2CN(C)CCN2C)C)=O)ncnc(C)c1Br CCCC(C)(C)C(=O)NCCC(N1CC=CCC1C(=O)OC)=O C1(CCC(=O)OC)CCc2ccccc2C1.c12ccc(cc1)CCS2 c1(C(C)C)ccoc1C(=O)NCC1CCN1C(=O)CCSCC(N)=O c1(C(N2CC(C3CN(C(=O)C(F)C4CCC4)CCO3)C2)=O)ccc2nc[nH]c2n1 N1(CCN(CCO)C(C2C(N(C)C)CCN2C(=O)NCC)=O)Cc2ccccc2C1 C(=O)(C(C)(C)C(=O)NC)N1CCC(NC(c2c(CC)non2)=O)(CO)C1 N1(C(C2(COC)CC2)=O)CC(C)CN(C(c2cc(OCC)nc(F)c2)=O)C(C)C1 Cn1nnc(CNC(c2ncn[nH]2)=O)c1C(N1CC2(CSC2)C1)=O N1(C(c2c(C)nccn2)=O)CCC2CC2(NC(=O)CSCCN(C)C)CC1 c1(NC(C2CCN(CC)C2)=O)cc2c(cc1CNC(C1CCCCC1)=O)OCCO2 c1(C(N2C(NC(C3(COC)CC3)=O)C=CC2)=O)ccc(-c2cn[nH]c2)cc1 Cc1nc(C(=O)N(C)CC2CCCN(C(=O)CC3CCC3C)C2)n(C)n1 C1(NC(c2cccc(C)c2)=O)CN(C(c2nn(C)nc2Br)=O)CCC1O N1(C(c2c(CCC)n[nH]c2)=O)CCC(C(=O)NCC2CCC(F)(F)C2)C12CCC2 C1(C(=O)OC)CCCCC1C(=O)N(CCC(C(C)C)NC(C1CC2CC2C1)=O)C CC1CC2(CCCC2)CN1C(=O)C=CCNC(C1CC(=O)C12CCC2)=O N1(C(c2c(C)ncn2C)=O)CC(CNC(c2c[nH]nc2C2CC2)=O)C(F)(F)C1 N(C(=NCc1ccc(OC(F)(F)F)cc1)NC1CCC1)Cc1cnc(C)o1 Cc1cc(C(=O)NC2CC2CNC(c2cc(CC(C)C)[nH]n2)=O)ccc1C1CC1 c1(C(=O)N(CC(C)CNC(=O)COCC2(F)CC2)C)coc(C(F)F)n1 C1(C(N(CCNC(C(C)C)=O)C)=O)(CNC(c2c[nH]cc2C)=O)CC=CC1 Cc1cc(C(N2CCC(CNC(C34CCCC3OCC4)=O)C23CC3)=O)c[nH]c1=N N1(C(C(CC2CN(C(CCOC(C)C)=O)C2)F)=O)CCCCN(C)CC1 Cc1oc(C2CC2)nc1C(N1CCC(N(C(=O)C(N)=O)CCO)CC1)=O c12ccc(cc1)[nH]c(=O)c2=O.c1(CCC(=O)NCC(C)OC)ccn(C)c1 N1(C(C2(COC)CC2)=O)CCOC2(CCCN(C(C3CCCC(C)C3)=O)C2)C1 N1(C(CCSCCCC)=O)CC2CN(C(c3onc(CC)c3C)=O)CCC12 c1(C(C)C)ccc(C(=O)NCC2(C)CCC(NC(=O)Cc3csc(S)n3)C2)nc1 c1(C(=O)NC(C(C)NC(=O)CCc2cncs2)C)c[nH]nc1-c1ccsc1 C(C(CO)(CO)NC(c1cnn(C)n1)=O)N(C(CC1C(C)C1)=O)C O=C(C1CCc2nccn21)NCCC1CN(C(=O)CCC2=CCCCC2)CCO1 C(=O)(C(F)CC(C)(C)C)N1CCC(CCNC(C=Cc2ncn(C)c2)=O)CC1 CS(=O)(=O)C1CCCCC1N=c1cccc(S(=O)(=O)NCCF)[nH]1 C12(C(N3CC(O)(CCNC(c4cccc(Br)n4)=O)C3)=O)CCC(CC1)C2 C=CC(C)(O)C(=O)N(CC(C)C(=O)N(CCCC)C)C C=CCC(C(=O)NC1COCC1O)NC(=O)Cc1ncccc1F c1(C(=O)NC(CC(=O)NC2(COC3CC3)CC2)C2CC2)cc(CCO)on1 N1(C(c2cn(C(C)(C)C)nc2)=O)CCCC(CNC(C2CCCC2(C)C)=O)C1 Cc1ccnc2sc(C(=O)N(C)CCN(C(=O)C3=C(Cl)CCC3)C)c(C)c12 N1(C(C2(OC)CCCOC2)=O)CCCN(C(=O)CCN2C(=O)CCC2=O)CC1C c1(C(N2CCC(N(C)C(C3(F)CCOC3)=O)C2)=O)cn(C)c2ccc(F)cc12 C1(CC(=O)NC)CCN(C(=O)CC=CCNC(C2(CCO)CC2)=O)C1 Cc1cc(Br)cc2cc(C(=O)NC3CN(C(C4COCCC4C)=O)C3)[nH]c12 C12(NC(C3CC(=C)C3)=O)CCOCC1CN(C(c1cc3c(s1)C(C)(C)CCC3)=O)C2 C1(O)(C(C)NC(C2(F)CCCC2)=O)CN(C(=O)CC2CSCCS2)C1 N1(C(C)C)CCC(C2CCCN(C(c3cncc(CN(C)C)c3)=O)C2)C1 N1(C(C=CCN(C)C)=O)CCC2(CCC2)C(NC(=O)C(C)(CC)OC)C1 N1(C(CC=C(C)C)=O)CCC2CCN(C(c3ccc4c(c3)C(=O)NC4)=O)CC12 c1(NC(C2CCN(Cc3cncc(OC)c3)C2)=O)ccc(C)c(OC)c1 c1(C(=O)NCC2(CO)CCN(C(C(C)S(N)(=O)=O)=O)CC2)cc(F)cc(F)c1F C(=O)(C(C)C(C)n1cccn1)N(C)CC1(CNC(c2nc(CCC)sc2)=O)CC1 c1(C(=O)OC)cc(=NCC2(NC(C3CCC4(CCC4)O3)=O)CCOCC2)[nH]cn1 c1(C(C(=O)NC(CC)C)N(CC(C)(C)C)CCOC)ccc(OC(F)F)cc1 S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)N1CCC(NS(=O)(=O)Cc2ccncc2)C1 c1(OCC)cccc(C(CO)NCC2COC(C)C2)c1 c1(C(N2CC(O)(CC(=O)OCC)C2)=O)c(NC(=O)C(C)CC(N)=O)sc(C)c1C Cc1cc(C(=O)N(C2CC(NC(=O)Cc3cc(C4CC4)on3)C2)C)c(O)nc1C O=C(CCCCCC1CC1)NCC1CCCN1C(=O)CCc1cncs1 C1(C(C)NC(C2(CSC)CC2(F)F)=O)CCN(C(C2CCC2)=O)CC1 c1(NCc2c(F)ccc(N)c2)cc(=NCC(=O)N2CCCC2)[nH]cn1 N1(C(CN(C(=O)OCC)CC)=O)CC(NC(c2ncc[nH]c2=O)=O)CC(O)C1 N1(C(C(=O)N(C2CCCCCC2)CC)CC(C)C)CCOC(C)(C)C1(C)C N1(C(c2c(N(C)C)cnc(Cl)c2)=O)CCC2(CCO2)CC1 Cc1nn2ccccc2c1C(=O)NC1CC1CNC(=O)CC1CCCNC(=O)C1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N(C(C1CC(=C3CC3)C1)=O)C2 C(=O)(C(C)C(F)F)N(C1CCCCCC1)C(c1cnc(CCC)s1)=O.C1C=CCS1 N#Cc1ccc(O)c(CN2CCCC(C(=O)NCCc3cnc[nH]3)C2)c1 C1(Cn2cc(CCCNC(=O)C(C)Cc3ccc(F)cc3)nn2)CC2CCC1C2 Nc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(-c3c4c(nn3C)CCC4)cc2)c1 CCC1=NOC(C(N2CCC(N(C(=O)CC(F)(F)F)CC)C2)=O)C1 C1(NC(C(C)Oc2ccccc2)=O)CN(C(c2cc(O)nc(Cl)c2)=O)CC1(C)C c1(C(CCCC)C)nc(-c2cnn(C)c2)nn1CCCn1ccnc1 c1(C(=O)NC2C(NC(C(C)O)=O)C2)cn(C)nc1-c1cccs1 c1(N(C)C)cccc(C(=O)NC2(CNC(=O)COCCF)CCCC2)n1 Cc1n[nH]c(C)c1C(=O)N(C1CCCN(C(=O)C(C)OCCC(C)C)C1)CCF c1(C(=O)NC2CC(CNC(=O)CC=C(Cl)Cl)C2)n[nH]c2ccccc12 N1(C(Cc2c(CC)con2)=O)CCCC(C(=O)NCc2cc(Cl)ccn2)C1C CN=c1nc(C(N2CC(NC(C3C(F)(F)C34CCC4)=O)C(O)C2)=O)cc(C)[nH]1 C1(COC)(NC(=O)CCC(C)N(C)C)CCN(C(=O)C(C)(C)c2ccccc2)C1 C(CC(C(=O)N1CC2CC1C2NC(=O)C=CCO)NC=O)SC CC(=O)CC(C)(C)CC(=O)N1CC(NC(=O)CC(C)(O)C2CC2)CC2(CC2)C1 C1(NC(=O)CC(c2ccccc2)C2CC2)CCC(NC(c2cccnc2S)=O)CC1 C=CCCC(CC(C)C)C(=O)N1CCC(C2(NC(=O)CC3CSCCS3)CC2)C1 Cc1ccc(CN2CCCC(CC(=O)NC3CC(F)(F)C3)C2)c(O)c1 N#Cc1ccnc(NC2CC2C(=O)Nc2cccc(O)c2Cl)n1 N1(C(c2cnc3ncnn3c2O)=O)CCCC2(CCCCN2C(=O)C(F)Cl)C1 C(=O)(C1=NN(C)C(=O)CC1)N1C(CNC(CCCC(=O)NCC)=O)CCC1 N1(C(C2(C#N)CCOC2)=O)CC(C(N2CCCC(O)(C(N)=O)C2)=O)C2(CCC2)C1 C(=O)(C(F)CCC(C)C)NC1C(C(=O)NCCC)CCCC1 N1(C(Cn2c(C(F)F)cc(C)n2)=O)CCC(C2(NC(c3cnc(S)[nH]3)=O)CC2)C1 c1(C(=O)NC(C(N2CC3(N(C)CC3)C2)=O)(C)C2CC2)cnn2ccc(Cl)c(F)c12 C1(CNC(C=C(COC)C)=O)CN(C(c2ccn(C3CCOCC3)n2)=O)C2CC12 N1(C(CC2CCN(C(Cc3cn(C)nc3)=O)C2)=O)CC(C(=O)O)CC(C(=O)O)C1 C(=O)(C(CCC1CCC1)NC(C1C=CC=CC=C1)=O)N1C(C)(CCO)CC1 c1(C(C)NC(CN(C(=O)CCc2ccn(C)n2)CCC)=O)ccnc(C)n1 c1(C(C(=O)NCC(CC)NC(C2(c3cnccn3)CC2)=O)C)cnccc1C CCC(C)CCCC(=O)NCCOCCCNC(=O)Cn1cc(C2CC2)cn1 CCCCCC(C)(CC)C(=O)NC1C2CCN(C(=O)C(C)(C)CC(F)F)CC12 c1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)C2)ncc(C#N)cc1Cl c1(SCC(=O)N(CCCC)CCCC)cccc(C)c1C.c12cccc(c1)C(=O)N2 Cc1cc(C)c(C(N2CCC(CNC(=O)C(S(N)(=O)=O)c3ccccc3)C2)=O)s1 c1(C(N2CC(NC(C3SC4C=CC3C4)=O)(CO)C2)=O)ccc(CO)cc1 C1(COC(=O)NCCCC)CCn2cc(-c3ccccc3C(F)(F)F)nc2C1 C1(NC(Cc2ccc(SC)cc2)=O)CCC2(CC1)CC2NC(=O)Cn1ncnn1 n1(CC(=O)Nc2ccnn2CC2CCCC2)ccc(=O)c2ccccc12 c1(C(N(CCNC(c2cc(OC)nn2C)=O)C)=O)nc(C)c(C)cc1N N1(Cc2n(C)nc(C3CCC3)n2)CCC2(NC(=O)C(=O)NC3CC3)CCCC12 N1(C(CC(CC)c2ccccc2)=O)CC(CNCC(F)(F)C(F)(F)F)C(C)(C)C1 C1(C(=O)NCC23CN(C(C(CCC)NC(C)=O)=O)C(C2)C3)(CC)CCC(F)(F)CC1 c1(OC)cc(C(=O)OC(c2ccnn2C)CO)c2c(c1)CCC2 c1(C(c2n(CCOC)nnn2)NC(C)C(C)C)ccccc1Br.C1(C)CC1 N1(C(CC23C(CN(C(C(CC=CCC)C)=O)C2)CC3)=O)CC2(CCN(C)CC2)C1 c1(CC(=O)NCC2CCN(C(C(C(C)C)F)=O)C2C)ccc(Cl)cc1F c1(NC(c2cn(CCC(C)C)nn2)=O)ccccc1C(N(CCO)CCO)=O CCC(C)(CO)C(=O)NC(CC1CC1)CC(=O)O.c12cn(nn1)C2C1CCC(=O)O1 N1(C(C23CC(C#N)(C2)C3)=O)CCC(O)(CNC(=O)CC2CNC(=O)O2)CC1 c1(CC)nc(=N)[nH]cc1C(=O)NCC1CN(C(=O)C(COC)CC)C(C)(C)C1 N1(Cc2c(C=O)cccc2)CCc2c(Cl)cccc21 c1(C(N2CCC(NCCCCCC)C(C)C2)=O)ccc([N+](=O)[O-])cc1 c1(OC)ccn2ncc(C(=O)NC3CC3NC(c3n[nH]c(C)c3F)=O)c2c1 C1(CC(=O)NCCCCNC(c2nc(C(C)=O)sc2)=O)CCCCCC1(F)F C1(CCNC(=O)CSC(F)(F)F)CCCN1C(=O)CCc1nncs1 c1(C(=O)NCC2(n3ccnc3)CC2)cccc2ccoc12.C1(OC)CC2N(C1)C2=O C(CCCCC(=O)NC1CC(O)CN(C(c2cccc(O)n2)=O)C1)NC(C)=O S(=O)(=O)(c1ccccc1)NCC(=O)NC(C1CCCN(C(=O)CCCC(N)=O)C1)C N1(C(C(C)Oc2cccnc2)=O)CCC(NC(=O)Cn2cnc(=N)[nH]2)C(C)C1 N1(C(Cc2nc(C)c(C)s2)=O)CCC(NC(C2(CF)COC2)=O)C(C)(C)C1 c1(OC)ccc(C(N2CCN(c3ccc(NC(=O)C=CCF)cc3)CC2)=O)nn1 N1(C(C(=Cc2ccco2)C)=O)CCC(C)(NC(c2ccn(C)c2)=O)CC1 N1(C(c2c(CC)non2)=O)CCC(C(C)C)CC1C(=O)NCCC(O)C(F)(F)F C1(N(C(C(C)SC(C)C)=O)C)CN(C(c2cnn(CCO)c2)=O)CC1(C)C C1(C(N(C2CC(O)C2)C)=O)CCC2CCC1N2C(=O)C=Cc1ccco1 N1(C(C2(CC=C)CCCC2)=O)C2CCC1C(C)C(NC(C1CCC(F)C1)=O)C2 C1(C(C)NC(c2c(OC)nsc2)=O)CCCN(C(=O)CCOCCN(C)C)C1 N1(C(c2nc3ccc(OC)cc3cc2)=O)CC(S(=O)(=O)CC(F)(F)F)C1 C(=O)(CCCC(=O)N(CCCCCC(=O)NC1CC12CC(O)C2)C)N(C)C N1(C(c2c(OC)cnnc2)=O)CC(CNC(C2(C)CCC2)=O)CC(C)C1 C#CCC(C)(C(=O)NCCOCCOC)NC(C1CCC2CC1CO2)=O Cc1cncc(C(=O)NC2(C)CC(C(=O)NCCC3CC4CCC3O4)C2)c1 N1(C(C2(COC)CCCCO2)=O)CCOC2(CCN(C(=O)Cc3cncs3)C2)C1 CCCC(C(=O)OC)NC(=O)NC1CCC(C(=O)OC)C1 N1(C(C2CCN(CC)C2)=O)CC2CCCC2C1C(=O)N(CCCC(=O)NC)C c1(COC(C(COC)OC)=O)cccc(F)c1 N1(C(C2(C=C)CCC2)=O)CCC2(CCCCN(C(=O)C(C)(C3CC3)OC)C2)C1 CC(C)(C)CCC(=O)NC(C1CN(c2ncc(C(F)(F)F)cc2Cl)CC1(C)C)=O c1(C(N2CC(C)C(CNC(=O)C3=CCCCCC3)C2)=O)[nH]cc2c1CCS2(=O)=O CON(CCC(=O)NCC1CCC2(CC2)CO1)C(=O)C1CCSC1 C1(C(=O)NCCN(C(c2n[nH]cc2F)=O)CC)CCCC1n1cccc1 N(C(=NCCCn1cccn1)NCC1CCOC1)CC1C(O)CCCCC1 c1(C(N2CCC(N(CCC)C(c3nncn3CC)=O)C2)=O)cc2sc(Cl)cc2[nH]1 N1(C2(C(C(C(=O)NC)(C)C)=O)CCC2)CCCC(C2CCCCN2)C1 c1(N(C)Cc2nccc(C)c2)ccc(S(=O)(=O)NCCC2CC2C)cc1Cl C1(C(N(CC(C2CCC2)OC)C)=O)CCCC1CNC(c1csc(O)n1)=O CC1(C)CC(NC(c2cc(Cl)ccc2N)=O)CN1C(C1CC2CCC(C1)O2)=O O=S(Cc1cccnc1Br)CCCCc1ccccc1 C(=O)(CCC(=O)N(C)C)N(CC)CC1CCCN1C(C1(C#N)CCOC1)=O c1(C(N(C(c2ccccc2)CNC(C(CC)C)=O)C)=O)cc2cccnc2cn1 C1(C)(CNC(CC2C(OCC)CN(C(=O)CC#N)C2)=O)CCCC(=O)N1 C(=O)(C(O)CC1CCOCC1)NCC=CCNC(c1conc1C(F)(F)F)=O C1(C(N2C(CN(C(Cc3c(C)ocn3)=O)C)CCC2)=O)Cc2nccn2C1 C1(NC(Cn2nc(C)oc2=O)=O)CC(C)CN(c2nnc(C(C)C)o2)C1 Cc1c(C(N2CCCC(N(C(=O)C(C)O)C)C2)=O)[nH]ccc1=O C(C(COC)CC(=O)NCC(O)CNC(c1ccc(F)cc1N)=O)OC C1(c2n(CCCOC)nnn2)(NCC2CCC(C)C2)CCC2(CCCCCC2)C1 C1(C(=O)NCC(CNC(C(C=C)O)=O)C(F)(F)F)CC2(C1)CC1(CC1)C2 c1(CC)[nH]c(=N)sc1C(=O)NC(C)CC(C)NC(=O)C=C(C)c1ccsc1 Cc1nc(NC(CN2CCCCC2)C(C)C)cc(N2CC(CF)C2)n1 N1(C(C2(C(=O)NC3CCCC3(C)C)CCCC2O)=O)C2CCC1CC(CO)C2.CC c1(CC)ccc(C(=O)NC2(CNC(C3CCN(C)C(C)C3)=O)CCOC2)cc1F c1(NCC(CC(C)O)C)nc(N2CCc3cncnc3C2)nc2sccc12 c1(C(C)CC(=O)N(C)CCN(C(=O)CCc2cc[nH]n2)C)ccc(F)cc1 CCC(C)CCCCC(=O)N1CCCC(NC(=O)COc2cccc(Cl)c2)C1C N1(C(C(C)OCC#C)=O)CCC(OCC(=O)NCCSc2nnc(O)o2)C1 N1(C(CC2CC(=C)C2)=O)CCCC1(C)CN1CCN(C(=O)CC2(OC)CC2)CC1 C1(C(=O)NC(C(C)(C)CO)CO)CCCCCCN1C(=O)CSC(F)F C1(OC)CC(CNC(C2(N3CCCC3)CCC2)=O)N(C(c2[nH]c(C)cc2C)=O)C1 CCN=c1[nH]cc(C(=O)NCC2CC3CN(C(C4(C)CCCCO4)=O)CC23)s1 n1(CC)nccc1C=CC(=O)N(CC(O)CN(C(=O)C(C)O)C)C C(CC(C)C(F)F)NC(CC(C1CC1)NC(COCCCC#C)=O)=O C1(NC(CSc2c(OC)cccc2)=O)COC2(CCN(C(C3CCC3)=O)C2)C1 c1(CC(=O)NC2CC(NC(C(CCC)=CCC)=O)C2)ccc(Br)c(O)c1 C(=O)(CCC(C)C(C)N1CCC(C(=O)NCC2CCCN2C2CC2)CC1)OC CCC(CC)C(C)C(=O)N1CCC(C(C)NC(=O)CCSC)C1 c1(NC(C2N(C(C3(CC#C)CCOCC3)=O)C3C(C2)C3)=O)ccc(C)c(Cl)c1 c1(C(=O)NCc2cc(C(=O)NC(c3ncnn3C)CC)on2)cn(C)c(C)n1 c1(C2(C(C)(C)C)CC2)cccnc1.C1CCCNC(=O)NC12CC2 C1(O)(CNC(=O)CCc2cnn[nH]2)CCN(C(c2c[nH]c(Br)c2)=O)C1 N1(C(C2CN(C(C)C)C2)=O)CCCC(C2CN(C(c3ccnnc3)=O)C2)C1 C(=O)(C(C)(O)C(F)(F)F)N(C(=O)Nc1cc(F)c(OC)c(F)c1)C c1(C(=O)NC(CCC)CNC(=O)CCc2ncc(C)[nH]2)c(C)cccc1O c1(C(N(CC(C)NC(c2cccc(CC)n2)=O)C)=O)cc(F)c(O)c(Cl)c1 N1(C(C(CC)C(C)C)=O)CC2CC(NC(=O)C(F)(F)c3ccnn3C)CC1C2 N1(C(CC(C)(C)C#N)=O)CCCCC2(C1)CN(C(=O)C(C)(C)C1CCC1)C2 N1(C(COCCC)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1C NS(=O)(=O)c1cc(C(=O)NCC2CCN2C(=O)CC2CCOC2)c(Cl)o1 N1(C(C2(C#C)CCC2)=O)CCN(C(c2cc(F)ccc2Cl)=O)C(CC(F)F)C1 c1(C(=O)NCC(CNC(CCC(=O)OC)=O)CO)ccc(OC)c(Cl)c1 C1(C(N2CC(CC(=O)NCc3cncc(Cl)c3)(OC)C2)=O)CC2C=CC1CC2 O=S(=O)(c1cccnc1NC1CC1)N1CCC(OC2CCC2)CC1 c1(C(C(=O)NC(C2CN(C(=O)CCOC3CC3)C2)C)C(N)=O)ccccc1 N(C1CCc2cccnc21)C(=O)NCCC(=O)N.c1(CN)ccccc1 C1(C(NOCCC(C)C)=O)COCCN(C(=O)C(c2cccnc2)C)C1 C(C(CC(C)C)NC(=O)CCCNC(=O)C1CC1)NC(c1c(CC)cco1)=O C12(C(=O)Nc3cnc(C)nc3)COCC1CN(C(c1ccc(F)cc1F)=O)C2 c1(C(=O)OC)cc(CC(N2CC=CC(NC(=O)C(C)OC)C2)=O)ccc1Cl N1(C(Cn2ccc(C)n2)=O)CC(C(=O)NCc2n[nH]cc2C)C(CCC=CBr)C1 Cc1[nH]nc(C(=O)NCCOC2CN(C(c3ccc(F)cn3)=O)C2)c1Cl C(=O)(C1=NOC(C)(C)C1)N1CC(C(C(N2CC(C)=C(C)CC2)=O)O)C1 C=CCCC(C(=O)NCC(O)CN(C)C)NC(=O)C(CO)OC C(=O)(C(Cc1ccsc1)C1(N(C2(C)CC2)C)CC1)OC=O.C1(=O)CN1.C(C)(C)(C)O N(C(=NCC1COCCO1)N1CCCC1)C(c1ccco1)C c1(C(N2CCC(C(C)NC(=O)CC3CC34CC4)CC2)=O)ccc(N)c(Br)n1 c1(CN2CC3(C(CC)C3)C2)nc(-c2ccc(C)cc2)c(Br)s1 C(CO)(C(C)NC(C1(Cl)CC1)=O)NC(C(C1CC1)SC)=O c1(C(=O)NCC(C)N(C(c2ccnc(C(C)C)n2)=O)C)c(N)cccc1Cl C1(CC)CCC(C(=O)NCc2ccccc2CNC(C2CCC(O)CC2)=O)CC1 C1(N2CC(N3CC(C)(CCC(N4C(C)COCC4)=O)C3)C2)C2CCC(C2)C1C.CO c1(C(=O)NCCCCN(C)C(C2CCS(=O)(=O)N2)=O)ccc(=O)n(CC(C)O)c1 C1(NC(Cc2nnc(C)s2)=O)CC2CN(C(=O)Cc3ccccc3C#N)CC2C1 C1(C(N(C2CC2)CC2N(C(C(C(C)C)C)=O)CCC2)=O)CC(F)(F)CCC1(C)C CC1(C)CCN(C(=O)C2=C(Cl)CCC2)C(C(N2CCCCC(F)(F)C2)=O)C1 Cc1ccc2oc(=NC3CCCC(NC(c4ccnn4CC(C)C)=O)C3)[nH]c2c1 C(=O)(C(C(C)C)n1ccnc1)N(CCCNC(C1COCCOC1)=O)CC C(=O)(CCCC(F)(F)CO)N1CCN(C(Cc2cnc(C)[nH]2)=O)CC1C1CC1 C1(NC(C=Cc2cc(OC)ns2)=O)CN(C(=O)C(C)(F)F)CC12CCOCC2 N1(C(c2c(CC)occ2)=O)CC(F)(F)CC1C(=O)NCCN1CC2CC2C1 c1(OC)ccc(CSC2CCC2C)c(-c2ccn(C)n2)c1.C1C(=O)O1 C#CC1CN(C(=O)COC2CN(C(=O)C(CC)NC(N)=O)C2)C1 N1(C(C=C(C)C)=O)CCC2(CC1)CC2NC(=O)CC(C)(C)C(=O)OC(C)(C)C C1(COC)(NC(=O)CCN(C)C)CCN(C(=O)C=CC(C)(C)SC)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)C(c2ccncc2)C)ccc2ocnc2c1 Cc1c(C(=O)NCC(c2ccccc2)CNC(=O)C(C)(C)CC#N)cccc1O N1(C(NOCC)=O)CCC(N2CCCC2C)CC1 c1(C(=O)NC2CC3(CN(C(c4c(C)nn[nH]4)=O)C3)OC2)ccc2[nH]nc(Cl)c2c1 CC1(O)CCC(CC(=O)NC2COCC2NC(=O)Cn2cccc(O)c2=O)CC1 CCC(C)(C)C(=O)C(=O)N1CC(NC(c2cnc(OC)nc2)=O)CC1C c1(CC)cc(C(N2CCC(NC(c3cccnc3CC(=O)OC)=O)C2)=O)n(C)n1 N1(C(CSC)=O)CC2(C1)C(NC(c1oc(C)nc1C)=O)CCS2(=O)=O C1(NC(c2c(C)ocn2)=O)CCCCC12CCN(C(=O)C(C)(C)C1CC1)CC2 C(C(C)CN=c1nc(N2CCCC(OC)CC2)cc(C)[nH]1)OCCOCC N1(C(C(COCC)n2cc(C3(C)COC(C)(C)OC3)nn2)=O)CCC2(CC(CO)C2)C1 N1(C(C2CC3(CC3)C2)=O)CC2(CCCN(C(=O)COCC(F)F)C2)C1 c1(C(N(C2C3CN(C(=O)C(C)(F)F)CC23)C)=O)ccc(CCC#N)cc1 CCC(CC(=O)NCc1nc(C(N2CCC(CCO)C2)=O)c(C)o1)OC c1(C(=O)NC2C=CCN(C(c3cc(F)ccc3F)=O)C2)cccc2c1CCC2 C1(NC(=O)C=Cc2cccc(Cl)c2)CCN(C(c2ccoc2)=O)CCC1CO C1(NC(c2ncccc2F)=O)CCN(C(c2ccc(-c3ccccn3)s2)=O)CC1 CCC(F)(F)CC(=O)NC(C12CCC(CC1)C2)CNC(c1cnoc1C)=O c1(CC(=O)NCCN(C(c2cc(CCC)[nH]n2)=O)C)noc2ccccc12 C(=O)(CCC(C)(C)C)N1C(C(C)NC(=O)CCOCC2CCOCC2)CCC1 C1(COC)CC(CNC(=O)Cc2csc(C)c2)N(C(c2nn(C)cc2C)=O)C1 N1(C(COCCC)=O)CCC2CN(C(C3CCN3C3CCCC3)=O)CC2CC1 C123COCC1CN(C2)C3=O.C1(C(=O)OC)CCC(NC(C2CCCC2C)=O)C1 C12(C(=O)NCC3CC3NC(C34CC3COC43CCC3)=O)CCC(O)(CC1)CC2 Cn1ncnc1-c1ccc(C(=O)NCCNC(=O)C(C#N)Oc2ccccc2)s1 N1(C(C2CCC(C(N)=O)C2)=O)CCCN(C(C2CCC(=O)N2)=O)CC1 C1(c2nc(-c3ccccc3)nn2-c2cccnc2)CC(C2CCCC2)C1 n1(CC)nc(C)cc1C(=O)NCC(=O)NC(C)CC1CCC1 c1(CCC(=O)N(CCCN(C)C(C2CCCCC2O)=O)C)cc2ccccc2[nH]1 CCC(C)CCCC(=O)NC1(C(=O)NCc2cc(C3CC3)no2)CC1 c1(C(=O)NCC2CCC(NC(C3C(C)(Br)C3)=O)C2)ccc(CO)c(Cl)c1 C(CC(C)(C)C)(C(=O)N1CC(C)CC1C(=O)N(C12CC(C1)C2)C)OC c1(CN(C(c2nc(CC)co2)C(=O)NCC=C)C2CC2)ccc(SC)cc1 C1(CC)CC(OC(=O)OC)(OC)C1.CCCCCCN1CCC(C(=O)NC)C1 C12(NC(CCOC)=O)CCCCCC1N(C(c1cc(Cl)no1)=O)CC2 C(=O)(C1CCCn2ncnc21)N(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)CC C1(C)(CC)C=C(C(=O)NCc2cccc(NC(=O)C(O)CN(C)C)c2)C1 c1(OC)ccc(C=CC(=O)NC(CNC(c2[nH]c(C)nc2C)=O)CO)c(OC)c1 C1(NC(C2CC23CCOCC3)=O)CCSC12CN(C(c1cnn(CCO)c1)=O)C2 Cc1nn(C)c(C(N2CCC(NC(c3ccccc3OC3CC3)=O)CC2)=O)c1F c1(C(N(CC(C)N(C(=O)CCc2ccn(C)n2)C)C)=O)ccc2nnn(C)c2c1 c1(C(=O)NC23CC(NC(C4C(C#C)C4)=O)C(OC2)C3)cc(S(N)(=O)=O)ccc1C c1(CCNC(C2CC(NCc3cn(C)nn3)C2)=O)ccc(C#N)cc1F C(=O)(C1CCc2cc(F)ccc21)N1CCCC(CN(C(=O)CC=C(Cl)Cl)C)C1 C1(NC(CCc2nc(C)c(C)o2)=O)CN(C(C2CCOC2C2CC2)=O)CC1(C)C N1(C(C=Cc2ncc(C)[nH]2)=O)CC(NC(=O)CCS(C)=O)CC(C)(C)C1 N1(C(C2(CC=C)CC2)=O)CC2CC(NC(C3OCCOC34CCC4)=O)C(C2)C1 C(=O)(CC(CNC=O)CC(C)C)N1CC(COC)N(C(=O)C(C)CCO)CC1 C1(NC(C2C3CN(C(C45CSCC4C5)=O)CC23)=O)CCn2cnnc2C1 C1(N(C(=O)CO)Cc2cccc[n+]2[O-])C2CC1CN(C(c1ccoc1Cl)=O)C2 c1(C(=O)NCCOC2CN(C(C(C)C3CCCO3)=O)C2)c[nH]c2ncccc12 CC1=C(C(=O)NC2CN(C(c3ccccc3C3CCC3)=O)CC2C)CCCC1 CC(C)CCCC(=O)NCCCC(=O)NCC#CC#CCO c1(C(=O)NC2CC(C)(NC(c3c(CC)[nH]c(=N)s3)=O)C2)cc2cc(F)ccc2s1 C(=O)(C(C(C)C)NS(N)(=O)=O)NCC1(C(=O)N(CCCN(C)C)C(C)C)CC(=C)C1 c1(SC)ccc(C(=O)NC2CCCC2CNC(=O)CN(C)C(C)C)cc1[N+](=O)[O-] c1(NC(C(N2CCOC2=O)C)=O)cccc(NC(C2CC(F)(CF)C2)=O)c1 C1(NC(Cc2ncc(CC)[nH]2)=O)(CNC(=O)Cc2ccoc2)CCCCC1C N1(C(C2(N(C)C(c3ccc(CO)s3)=O)CC2)=O)CC2CC(CO)C(C2)C1 c1(C(N(c2nccn2C)CC)=O)sc(Br)cc1I c1(CC(=O)N(C2CCN(C(C3CCN(C)C3)=O)C2)CC)cn(C)nc1C C=C1CCC(C(=O)NC(C2(O)CN(C(=O)C(C)OC)C2)C)CC1 CCC(CCCC(=O)N1CCCN(CC)CC1)NC(=O)CC1CN(C(C)=O)C1 c1(CN2CC(C(C)NC(c3cnoc3-c3cnn(C)c3)=O)C2)ncn2ccccc12 C(N=c1nc(CC2CCCOC2C(C)C)c2c([nH]1)COC2)C1(SC)CCCC1 C1(C(=O)NC2(CNC(CCOC(C)C)=O)CCCCC2)CCCC2(C1)CC2(F)F C1(CNC(C(C)OC2CCCC2)=O)CC12CCN(C(=O)CCCC1CC1)CC2 C(=O)(C(C)(F)C(F)(F)F)NC1C(C)(C)CN(C(c2ccc(Br)cn2)=O)C1 C(CCNC(C1(CCOC)CCOCC1)=O)(C(C)C)NC(CCCC)=O C1(CC(N2CC(C(N)=O)(CNC(c3n(C)ccn3)=O)C2)=O)CCC(F)(F)C1 C1(NC(CN2CCN(c3cc(C)ncn3)CC2)=O)CC(=O)N(C)C1c1cnn(C)c1 CC1(C)CCCN(C(C2CC3(C2)CC32CC2)=O)C1C(=O)NC1(c2nc[nH]n2)CC1 Cc1cc(C(=O)NCC(Cl)(Cl)Cl)cc(C)c1C#N c1(NC(=O)OC(CCN(C(C)=O)CC#N)=O)cccc(F)n1 c1(C(N(C2CCN(C(C3CCSCC3)=O)C2)C)=O)cncc(N)c1 n1(CC)ccc(=NC(=O)C2CC(O)CCN2C(=O)C2=CCSC2)[nH]1 Cc1nc(C(C)C)[nH]c(=NCC(C2CC2)NC(c2csnn2)=O)c1Br c1(C(N(CCCN(C(=O)CC2CCCN2C2CC2)C)C)=O)cccc[n+]1[O-] c1(C(=O)NCC(C2CC2)NC(C(C)(C2(C)CC2)OC)=O)cccc(Cl)c1 C1(N(C(C(C=C)OC)=O)CC2CC2)CCCN(C(=O)CC=CC)C1 c1(NC(CCCC(=O)NC)=O)ccc(-n2cc(C3CC=CCC3)nn2)cc1 c1(CC(N2CCOC(CCNC(=O)C(F)(F)CO)C2)=O)ccc(Cl)cc1F c1(C(=O)NC(CNC(c2c(CC)csc2)=O)(C)CC)cc2c(o1)CCCNC2=O c1(SC)nc(Cl)cc(=NC(C)CC2CC2)[nH]1.C1(=O)CCC(=O)N1 C1(OC)CCCCC1C(=O)NCC(O)CNC(=O)C(C)(C)OCc1ccccc1Cl C1(C)(COC)CC(NC(c2cnc(O)c(C)c2)=O)CN1C(=O)CC1CC(C)=NO1 C1(C(N2CCCC(CC)(NC(=O)C=Cc3ccoc3)C2)=O)CC12CCCCCC2 CCCCC(C)(F)C(=O)N1CCC(NC(c2cc3occc3[nH]2)=O)C(CO)CC1 c1(C(c2n(CCSC)nnn2)NC2CC2C2CCC2)ccc(F)c(C(C)C)c1 C1(C(NOC(=O)C(c2ccnn2C)C)=O)CCOC1CN.CCCCNC(=O)C c1(C(=O)NC2CCN(C(C3CC(CC)C3)=O)CC2)ccc(S(C)(=O)=O)[nH]1 c1(COC)ccc(C(=O)Nc2nc(C(c3ccccc3)O)cs2)c(Cl)c1 C(=O)(C(O)CC[S+](C)C)NC1CC2CN(C(c3cccc(C)n3)=O)C1C2 C1(C(=O)NC(C)C(C)(C)NC(c2cccc(=S)n2O)=O)CC2CC1CC2O Cc1sccc1CC(N1CCC1C(=O)NCCSC(C)(C)C)=O N1(C(C2CCC(C)(C)C2)=O)CCCC(F)(CNC(=O)CCn2cnccc2=O)C1 c1(OC)c(C(C(C)C)NC(=O)NC2(CO)CC=CC2)cccc1Br c1(CC)nnc(O)c(C(=O)NC(C)CCNC(C2COCC(C)(C)O2)=O)c1CC C1(N(C(=O)CC(F)F)C)CCCN(C(c2conc2C2(C)COC2)=O)C1 C(=O)(CC(C)C(=O)OC)NC1(COC)CN(C(c2ccccc2OC(F)F)=O)C1 C=CCC(C)(C)CN=C(NCc1ccc2sccc2c1)NCC(C)(C)C c1(OCC=C)ccc(C=CC(=O)NCCC2CCCCC23CC3)cc1F c1(CC(=O)NCC=CCNC(CC2(OC)CCCC2)=O)coc2cc(Cl)ccc12 C(=O)(CC1CCc2ccccc21)N1CC=C(CCNC(C2CC3CC2C3)=O)CC1 c1(C(=O)NC(c2ccccc2)C(C)NC(=O)C=C2CCC2)ccn(C)c(=O)c1 c1(SCC(=O)NC(C(=O)NC(C#C)C(C)C)CN(C)C)ccc(C)c(C)c1 c1(C(N2CCOCC(NC(c3c(C)nccn3)=O)C2)=O)n[nH]c2c1CC1CC21 CCCC(C)(O)C(=O)NC(C)CN(C(=O)COc1ccccc1CC)C C12CCC(CC1)C(=O)N2.C1(C(=O)Nc2c(C)scn2)C=CC=CC=C1 C1(C(C)C)CN(C(=O)C=CC=C(Cl)Cl)CCN1C(c1cn(C)nc1Br)=O c1(CC)ccccc1-n1cc(C(=O)NCCC(C)NC(=O)CCC2CCC2)nn1 N1(C(C2C(C)(C)CCO2)=O)CC2(CCCC(CNC(C3(C4(C)CC4)CC3)=O)O2)C1 C1(CCNC(c2ccns2)=O)(NC(CC2N(C)CCC2)=O)CCOCC1 S(=O)(=O)(c1cccc(C(F)(F)F)c1)NC1CCN(C(C2(CO)CCC2)=O)C1 N1(C(C2C3(CC(OCC)C3)C2)=O)CCCC2(CCN(C(c3n[nH]c(=N)[nH]3)=O)C2)C1 C1(NC(CC2(C)CCCCC2)=O)CC2CCC(C1)N2C(=O)C=Cc1ccncc1 Cc1ccc(F)c(COC(c2cccc(-c3ccc(Cl)cn3)c2)=O)c1 c1(C(N(C)CC2CCCN(C(CSCC=C)=O)C2)=O)ccc2c(ccn2C)c1 Cc1ccc(NC(c2cc(F)ncc2NC(c2ccc(Cl)c(I)c2)=O)=O)cc1F C1(NC(Cc2c(C)n(C)nc2)=O)CCN(C(=O)C=CCn2cncn2)C1(C)C c1(OCC(C)C)cccc(C(=O)NC(C)CCNC(=O)CC(C)C#N)c1 C(=O)(C#CC1CCOCC1)N1C(CNC(c2c(C)ccc(F)c2)=O)C(C)(C)CC1 CC1CN(C(C2(C)CCN(C)C2)=O)CCC1C(=O)N(C)CC1CN(C)C1 c1(-c2cccs2)ccc(NC(C2CC2)=O)cc1F.C1(C(=O)NCC)(COCC)CC1 C1(CCNC(CCSC)=O)C=CCN(c2cc(C)ncn2)C1 N1(C(c2[nH]cnc2C)C(=O)NC2CC(CC)C2)CCC(N2CC=CC2)CC1 N1(C(c2ccc(O)cn2)=O)CCN(Cc2ccc(N3CCCC3)cc2)C2CC12 c1(C(N(C(CNC(C(CC)(C)OC)=O)C)C)=O)ccc2nccc(C)c2c1 N1(C(C(CC=C)NC(C)=O)=O)CCC(F)CC1C(=O)NC(c1[nH]c(C)nc1C)C Cc1ccc(C(=O)NCC2CCC(C)CN2C(=O)COCC(F)(F)F)c(C)c1 C1(CNC(C2(C(N)=O)CC2)=O)CC(C(=O)NCc2cccc(O)n2)=NO1 N1(C(C(C(CC)O)(F)F)=O)CC=C(CC(=O)NC(c2nccs2)CC)CC1 CC1CC(=O)NC(C(=O)NCCC2CN(C(=O)CCOc3ccccc3F)C2)C1 c1(NC(c2nnnn2CC2CCOC2)COCC)ccc(OC)c(Br)c1 C=CCC(C(=O)N1CCCC1C=CC(N1CC(COc2ccco2)C1)=O)OC c1(C(N2CCC(O)(CC)CC2)C(=O)NCCOCC)ccc(=O)n(C)c1 C1(O)(C(N2CC(C3(NC(C4C(C)C4C)=O)CC3)C2)=O)CCCC(C)(C)CC1 C1(C(N2CC3(C(NC(CC(C)n4cccn4)=O)CC3)C2)=O)CC2(C1)CS(=O)(=O)C2 C1(C(=O)NCC(C)OC)CC2CCN(Cc3ccc(O)c(CO)c3)CC12 C(=O)(CC(=O)NCC(Cc1ccccc1)N(C(C12CC(F)C1C2)=O)C1CC1)OC O=C1Nc2c(C(N3CCC(Nc4ccc(F)cc4[N+](=O)[O-])C3)=O)cccc2C1=O c1(C(N2CCN(C(c3c(C)cc(N)cn3)=O)CC2)=O)cc2cccnn2n1 C1(C(=O)NC(c2nncn2C)CC)CC(F)CN1C(c1ccc[n+]([O-])c1)=O CC1=CC(C(=O)NCCOCCNC(=O)COC2CCOC2)SC1 c1(C(=O)NC2CCN(C(C3CC34CC4)=O)C2)n[nH]c(C2CC2)c1Br Cc1ccccc1-c1ccc(Cn2cnc(-c3ccncc3)n2)cc1 C(=O)(C(F)C(F)(F)F)NC(C(=O)N(C1C(C)C1)C)CO CCCCC(C)(F)C(=O)NC1CCOC1C(=O)NC1CCCC1 CC(C)C1=CCC(NC(=O)C(C)(C)C(C)NC(=O)CCC2CC2(C)C)CC1 c1(C(C)=O)cc(C(N2CCOCC2CNC(=O)C=CC(=O)NC2CC2)=O)n(C)n1 c1(C(=O)NCC=CCNC(c2c(-c3nc(C)sc3)c[nH]c2)=O)cc(F)cc(F)c1N N1(CC(=O)NCC2CCCC(NC(C3(C(N)=O)CCC3)=O)C2)CCCCS1(=O)=O N1(C(C2N(CC)CC2)=O)CC2CCC(CNC(c3c(C)cnn3C(C)C)=O)C2C1 N1(C(CCSC)=O)CCC2(CC1)CCN(C(C1CC(C)(C)OC(C)(C)C1)=O)C2 c1(-n2cc(CC3(NC(=O)NCC(CC)CC)CCCSC3)nn2)ccc(C)cc1 C(=O)(C1=CC2CC=CCC12)N1CC(CCNC(c2nnsc2C)=O)(OC)C1 C1(C(N2C(CN(C(COC)=O)C3CC3)CCC2)=O)C(C2CC2)C1(F)F c12ccc(C(N)=O)cc1NC(=O)C2.C12(CC1)C(=O)NCC2.C(=O)(C1CC1)OC.CS c1(C(=O)NC(C)CCCNC(C2CCCN2C)=O)[nH]c(=N)ccc1Br CC1(C)CN(C(c2ccnc(Cl)c2F)=O)CC(CNC(C2C3CCC(=O)C23)=O)O1 C(CC(CNC(=O)CCCc1cccs1)NC(=O)C(C)NS(C)(=O)=O)OC CN1N=CC(CC(N2CCC(OCC(=O)N(C3CCOCC3)C3CC3)C2)=O)C1=O C1(NC(C(C)O)=O)CCC2(CC1)CCN(C(C1CCCN1S(C)(=O)=O)=O)CC2 c1(C(=O)NCC2(COC)CN(C(C3CC(SC)C3)=O)C2)cnn(C)c1SC N1(C(C(C2(O)CN(C(c3c(C)coc3)=O)C2)F)=O)CCCC(N(C)C)C1 c1(-n2cc(C(=O)NC3CCN(CC)C3)nn2)ccc(C)cc1F CCC(CC(C)C)C(=O)N1CCOCC1CN(C)C(C1(OCC)CCOCC1)=O Cc1nn(C)cc1CC(=O)N(CCCNC(c1ncoc1C1CC1)=O)CCO c1(CC)scnc1C(=O)NCC1(C(=O)NCc2ccon2)CC1 c1(C(N2C(CNC(C(C)(C)OC)=O)CN(C)CC2)=O)ccc2nc(O)n(C)c2c1 c1(C(N(CC(CN(C)Cc2ccc(Cl)cc2Cl)O)C)=O)cncc2ccsc12 C(=O)(C(CCc1ccccc1)N1CCOC(CCO)C1)NC(c1cccs1)C C12(C(=O)NC(C3CCCCC3)CNC(C(CC)SC)=O)CCC(N=[N+]=[N-])C1C2 c1(OC)cc(CN2CC3(CC3)CC2C(=O)NCc2cc(Br)ccc2Cl)cc(Br)c1 c1(N(C)CCOCCN(C(=O)C(C)NS(C)(=O)=O)C)ncnc(Cl)c1C#N C1(NC(CC(=O)NCC)=O)CN(C(=O)CNC(c2cnoc2C)=O)CC(F)(F)C1 c1(C(N2CCCC(NC(c3cc(C)c(F)cc3)=O)C2C)=O)ccc(S(N)(=O)=O)o1 C=CC(C)CC(=O)N(CC(C)N(C(=O)C(F)CC1CCCC1)C)C N1(C(c2ncn(CCNC(=O)C=Cc3cn[nH]c3)c2)=O)CCC2(CC1)CC(O)C2 c1(C(C)=O)ccc(C(=O)NCC2CCC2NC(C2(C(C)(C)C)CCC2)=O)o1 C#CC1CC2CCC1N(Cc1cccc(NCc3ccc(F)c(C#N)c3)c1)C2 c1(C(=O)NC)ccc(NC(C23CC2CN(C(c2cccc(I)c2)=O)C3)=O)cn1 CC(C)(CC1CCCCC1)C(=O)NCC1CCCCN1C(c1cc(CF)on1)=O Cc1c(CCCC(=O)N(C2CN(C(=O)CC3(O)CC3)C2)C)cnn1C.C1(=O)CO1 n1(CC)cc(Cl)cc1C(N1CCC(C)(CNC(=O)COCC2CCOC2)C1)=O C(=O)(CC(C)(C)CNC(c1cc(O)cs1)=O)NCC(C(C)C)(C)C C1(C(N2CC3(C2)CN(C(C2CCC=CCCC2)=O)C3)=O)CCn2nnnc2C1 c1(C(N2C(C(C)NC(Cc3ncc(C)[nH]3)=O)CCCC2)=O)ccc2nnnn2c1 N1(C(C=CC(C)=O)=O)CCC(C)N(C(c2csc(C3CCCO3)n2)=O)CC1 C(=O)(CCC(=O)N(C)C)N(CCOCCN(C(C1CN(C(C)C)C1)=O)C)C CC(C)CC(C(=O)NCC1CCCS1)NC(C1CN(C2CCC2)C1)=O N1(C(c2cc(CCOC)on2)=O)CC2CCC1C(NC(C13CCC(CC1)C3)=O)C2 CC1CN(C)CC(C(N2CC3CC(CNC(c4ccc(N)c(N)n4)=O)C3C2)=O)O1 c1(-n2ncc(C)c2)ccc(C(=O)NCC2(NC(c3cscn3)=O)CCCC2)cc1 C(CCCC(C)(C)C(=O)NNC(=O)C1CCCS1)NC(C1(N(C)C)CC1)=O CC(CCCNC(=O)CCCn1cc(C2CCCO2)nn1)C(=O)O C1(CN(C(C(C)Cn2cccn2)=O)C)COCCN1C(=O)C=Cc1ccc[nH]1 C1(C(N(C2CC(NC(=O)CC3(C(F)F)CC3)C2)C)=O)CCC(=O)O1 N1(C(c2cc(C)sc2C)=O)CCC(F)(CNC(=O)CNC=O)CC1 c1(Cn2cc(-c3n(C)nc(C(F)(F)F)c3)nn2)cc(F)c([N+](=O)[O-])cc1F c1(C(=O)NCC2(N(C(=O)COCCc3nccs3)C)CCC2)ncccc1N c1(C(=O)NC(C)CNC(c2cc3c(ncn3C)s2)=O)ccc(F)c2cccnc12 C(=O)(C(C)CC(C)(F)F)N1CC(CCC)N(C(=O)C(=O)NCC2CC2)CC1 N1(C(C2C(C)(C)C2(F)F)=O)CCOC(C(=O)NCCOCCC2CC2)CC1 N1(c2nnc(CC)n2CCn2cnnn2)C2CCCC1CNC2 CC(C)(CCCCNC(=O)CCCOc1ccccc1)NC(C1CCC2CC12)=O c1(C(N(C)CC2CN(S(CC)(=O)=O)C2)=O)c(OC)ccc(Cl)c1F N1(C(C2C3CCCC23)=O)CC2(C(N3CC4(C3)CC4(F)F)=O)CCC1CC2 CN1C(=O)CN(CC(C(=O)C(c2ccc(Cl)cc2)F)=O)CC1=O.OC(F)F C1(C)(CNC(CCCC(C)=O)=O)CN(C(=O)Cc2nn(C)cc2Cl)C(C)(C)C1 CC1CCCCC1OCC(=O)NCCCC(C)(C)NC(=O)Cc1cocn1 c1(CC(=O)NC2C(NC(C3C(C)(C)C3)=O)CCOC2)ccc(Br)cc1F C1(NC(C(C(C)O)C)=O)CS(=O)(=O)CC1N=c1ccnc(C2CC2)[nH]1 c1(CNCCS(=O)(=O)NC2CCCC2)ccc(OC(F)(F)F)nc1.C1(N)CC1 N1(C(c2c(OC)csc2)=O)CCC(CC(=O)NCCOC)CC1 C1(C)(CNC(C(CC)Oc2cccc(C)c2)=O)COCCN(C(=O)C=CSC)C1 C(=O)(CCC(C)C)NCC(C1CC1)NC(C1CC(OCC)C1)=O Nc1ccc(S(N)(=O)=O)cc1C(=O)NCC1CCCN(C(=O)C(O)C(F)(F)F)C1 C#Cc1cc(C(=O)NC(CC(C)CC)C(=O)Nc2csnc2C)ccc1C C(=O)(CC=C(Cl)Cl)NC1(C)CC(NC(c2[nH]cc(C(C)(C)C)c2)=O)C1 Cc1ccc(C(N2CCOCC(O)C2)C(=O)NCC(C)C)c(Br)c1 N1(C(=O)COC2(CN)CC2)CC2(CC(NCC(C)OCCOC)C2)C1.OC c1(C(=O)NCC2(C)N(C(C(C=C=C)C)=O)CCC2)cc(C)cc2c[nH]nc12 C1(C(=O)NC2CCN(Cc3ccccc3)CC2O)CCn2c(O)nnc2C1 N1(C(c2cc(C(=O)OC)on2)C(=O)NCCC)CCCCC12CCOC2 CC(C)CC(O)C(=O)N(C1CCN(C(C2CC(O)CN2C)=O)CC1)C C1(CC(=O)NOCCF)CCCC(NC(=O)CC2CC(=O)NC2=O)C1 c1(C(=O)NC2CCCC(CNC(CC=CC=C)=O)C2)ccc(Br)c(C)c1 c1(C(N2CC(CNC(CSS(C)(=O)=O)=O)OCC2)=O)ccc2snnc2c1 c1(C(=O)NCC(Cn2cc(C(C)(C)O)nn2)(F)F)cc2ccc(Br)cc2cn1 C#Cc1ccnc(NC(N2CC3(C2)CN(C(=O)COc2cccc(Cl)c2)C3)=O)c1 c1(CNC(N(C)C)=O)ccc2c(c1)CCCC2NC(c1cncnc1)=O c1(CN2C(C(=O)Nc3cnc(C)c(Cl)c3)CC3CC32)c(F)ccc([N+](=O)[O-])c1F C(=O)(C1CCCc2nncn21)NCC1CN(C(C(C(C)O)N(C)C)=O)C1.C1CC1 CCN(OC)C(=O)C(C)N(C)C(C1(F)CC=CCC1)=O c1(C(=O)NC2(CO)CCN(C(C3COCCO3)=O)CC2)cccc2scnc12 Cc1ncnc(NCC2(C(N)=O)CN(C(C3CCN(C)C3=O)=O)C2)c1F NC(Cn1cccn1)C(=O)NCC1OCCO1 N1(C(Cc2c(C)nsc2)=O)CCC2CN(C(=O)CC3(C)CCOCC3)C2C1 C1(CNC(C2C(C(=O)OC)C2(C)C)=O)CC2(CO1)CN(C(c1cnco1)=O)C2 C(=O)(C(C#N)C(C)C)NC(CCC=C)C(=O)NC(C)CCSCC c1(C(=O)OCc2c(-c3ccc(OC)cn3)cccc2)cccc(Cl)c1Br N1(C(C(COC)C)=O)CCN(C(c2[nH]nnc2C2CC2)=O)C2CS(=O)(=O)CC12 c1(CC(=O)NC2CC2NC(=O)C(F)(F)Sc2ccc(F)cc2)c[nH]ccc1=O N1(C(C2C(C(=O)OC)C2)=O)CC2CC1C2NC(=O)CCc1ccncc1 CC(C)(C)C1=NOC(C(N2CCC(F)(CNC(C3C4CCC3CC4)=O)C2)=O)C1 C1(C)(C(=O)NCC#CCNC(C(=Cc2ccncc2)C)=O)CCOC12CC2(F)F C(C(CC(=O)N1CCC1)C1CC1)NC(C1(COC)CCC1)=O N1(C(c2occ(C)c2)=O)CCCCC(CNC(c2cc(C(=O)O)c(F)cn2)=O)C1 c1(C(=O)NC2CN(C(C3CC(SC)C3)=O)CC2CC2CC2)ccnn2ccnc12 C1(CC(=O)NC)CN(C(=O)CNCc2ccsc2)CCN1C(=O)CC(C)C(F)F n1(CCC(=O)NC2(C)CC(NC(CCC(C)OC)=O)C2)ccc(O)nc1=O c1(C(N2CC(NC(c3ccc4nncn4c3)=O)C3C2C3)=O)cc2ccccn2n1 C(=O)(C(O)CC(C)(C)C)N1CCN(C(CSCCCC)=O)CC1C(F)F c1(CNCC#C)cc2c(cc1F)NC(=O)CC2 c1(N(C)C)nc(Cl)c(C(=O)NCC2(CNC(=O)CC3CCCS3(=O)=O)CCC2)s1 C(=O)(C(CCCC)C1CCC1)N1CC(C(NOCCC(=C)C)=O)C1 C12CN(CCC1F)C(=O)c1c(cccc1F)-c1ccc(s1)-c1nccn12.CC C1(CC(=O)NCC(CNC(C=C(C)C(F)F)=O)CO)CCCC(C)O1 n1(CCN(c2ccc(OC)cc2C)C(C)(C)C)ccc(=NC(=O)NC(=O)C(F)F)[nH]1 N1(C(C2(CC)CCOCC2)=O)CC2CC(NC(C3CC(=O)NC3(C)C)=O)C2C1 N1(C(c2n(C)ncc2I)=O)CCCC(O)(c2cn(-c3cncc(F)c3)nn2)CC1 CC1CN(C(=O)C(c2cccnc2)O)CCC1CNC(c1ccncn1)=O c1(C(N2C3C(NC(C(C)OCCN(C)C)=O)C(C3)C2)=O)cc(S(N)(=O)=O)n(C)c1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NC(c1ccnn1C)CC)CCSC C#CC1(C(=O)NC2CCN(C(=O)CCCn3cccn3)CC2CO)CCCCC1 C1(CCNC(c2c(C)snc2)=O)CCCCN1C(=O)CSc1cccc(Cl)c1 C=C(C)C(C)(O)C(=O)N(CCCNC(=O)CCC1(C)NC(=O)NC1=O)C(C)C C(=O)(C(C)C(C)NC(=O)CN(C(=O)COCCCF)C)NCC CC1CC(NC(C2CC3CCCC23)=O)CN1C(=O)C(c1ccccn1)O Cc1cc(F)c2c(c1)CCN(C(=O)C(F)C1CCN1)C2 C1(C(N2CCC(Br)C2)=O)CC2OCCC2N(C(c2ccc3occc3c2)=O)C1 Cc1cc(C(=O)NCC2(Cn3cc(CCN4CCOC4=O)nn3)CC2)cc(C)n1 N1(C(COCCCC)=O)CC(F)CC1C(=O)NCCCCC(=O)NC C(C(C)(O)CNC(C1CCOC1CNC(=O)CNS(C)(=O)=O)=O)SC C12(NC(Cc3c(Cl)cn(C)n3)=O)COCCC1CN(C(c1cn[nH]c1)=O)C2 C(=O)(C(CC(C)CC)NC(=O)CN(C)C(C)=O)NC(CC#C)C(N)=O Cc1nc2ccc(C(=O)NCCCCNC(c3cc4cccnn4n3)=O)cc2o1 C(=O)(C(CNC(C1(Cl)CCCO1)=O)CC(C)C)NC(c1c(C)n[nH]c1C)C N1(C(C(C)OCC#C)=O)CCC(NC(c2cnn(C3CCCC3)c2)=O)C1C1CC1 N1(C(CC(c2cccc(C(F)(F)F)c2)NC(C(C)O)=O)=O)CCCC(N=[N+]=[N-])C1 O=S(=O)(c1c(F)cc(Cl)cc1F)NC1CCCN(C2COCC23OCCO3)C1 CC(CC(=O)N(CCCNC(C12CC(C)C1C2)=O)CCO)c1ccccc1 N1(C(=O)NC(C=O)Cc2ccccc2)CCC2(CCOCC2)CC1.CNC C1(C(=O)NC(CCCC=C)C2CC2)CC(N=[N+]=[N-])CN1C(c1cc[nH]n1)=O C1(Nc2sc(SCC)c(Cl)n2)CC2C3C=CC(C3)C12 c1(OCC)c(F)ccc(C(=O)N(CCNC(C2C3CCOCC23)=O)C2CC2)c1F N1(C(C(CC)=CC)=O)CC(NC(c2ccc(OC)s2)=O)C(C)(C)C1 N1(C(C23OC(C)C(C2)C3)=O)CCC2(CC1)CCN(C(=O)CCC(F)(F)F)CC2C N12CCC3CN(CC3CC1)CC2.C1(CCNS(C)(=O)=O)CNC(=O)CO1 c1(C(N(CC(C)N(C(Cn2c(C)nnn2)=O)C)C)=O)cc2n(n1)C(C)CCC2 C(C(N=[N+]=[N-])C(=O)NC1CCCC1C(=O)NC1CCCCCC1CO)OCC N1(C(c2ccc(CCCC)cc2)=O)CCC(NC(=O)C(C)=CC2CC2)C(O)C1 c1(C(=O)NCCCN(C(=O)Cn2cc(C3CC3)cn2)C)cc(F)c2[nH]nnc2c1 c1(C(=O)OC)cc(CC2CC2)no1.C12CCC1NC(=O)C1(CC1)CC(=O)N2 c1(C(=O)NC2(C)CN(C(c3nncc(C)c3)=O)C2)ccc2ccn(C)c2c1 c1(-c2cn(CC(CNC(C(C)CN(C(=O)CO)C)=O)(C)C)nn2)ccc(F)cc1 c1(C(=O)NC2C(NC(CSCCC=C)=O)C2)cc(COC)no1 Cc1cccnc1CC(=O)NCC1(C(=O)N(CCCCO)C)CCCC1 C1(C(=O)NC(CSC)(C)CO)CC(F)(F)CN1C(c1cncc(C#N)c1)=O CCC(CC)C(=O)NCCCCN(C)C(C1C2CCCC12)=O c1(C(=O)NC2CCC(C)N(C(=O)Cn3ncn(C)c3=O)C2)cc2n(c1)CCCC2 C1(NC(c2ccc(CC)cn2)=O)CC(OC)CN(C(=O)Cn2cnc(C#N)n2)C1 C(=O)(C(C)C(C)n1cccn1)NCCN(C(c1csc(C)c1N)=O)CC c1(OC)ncccc1NCCOCC(=O)NCC(=O)OC(C)C C(=O)(CC(C)CC(C)(C)C)N1CC(C(=O)Nc2cn(CC)nc2)C(O)CC1 CC1CC(NC(=O)COCC(F)(F)C(F)F)CCN1C(c1ccsc1)=O C1(CCF)(CNC(=O)CCNC(=O)CC2CCCOC2)CCOCC1 c1(C(=O)NC(C2N(C(c3n(CC)cnn3)=O)CCCC2)C)cc(C)c(C)c(C)c1 Cc1c(C(=O)NCC2CCC(F)(CNC(C34CCC(CC3)C4)=O)C2)ncn1C C#Cc1ccc(CC(=O)N(CCCNC(c2c(C)ccnc2Cl)=O)C(C)C)cc1 C(CN=c1[nH]c2cc(Cl)ccc2s1)OCCN(C(=O)CN1C(C)CCC1C)C(C)C Cc1ncccc1CCC(N1CC2CC2(CNC(C2CCSC2)=O)C1)=O N1(C(c2n(OC)cnc2C)=O)CCCCC(NC(C2CCN(C)C(=O)C2)=O)CC1 O=C(CCCCCO)NC(C12CC(CCN3CCS(=O)(=O)CC3)(C1)C2)=O CN1CC2(CCN(C(=O)CC3C(NC(c4nocc4Cl)=O)CC3O)CC2)C1 c1(N2C(C(C)(C)NC(C34CC3COC4(C)C)=O)CCCC2)cnc(C#N)cn1 c1(C(=O)NCC#CCNC(c2c(C(C)C)onc2)=O)ccc(F)c(C2(C)CC2)c1 CC1(C)COCC1.C1(CC(=O)NCCCNC(=O)OC(C)(C)C)CCCCC1S CC(CC(C)(C)C)C(=O)NC1(C)CC(NC(=O)C(c2ccc(C#N)cc2)C)C1 N1(C(C2(CC#C)CCC2)=O)CC(NC(C2CC(C#N)C2)=O)C2(CCC2)C1 N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(=O)C=CC(=O)N(C)C)CC2)C1 c1(C(=O)NCC2CCCCCO2)c(F)cc(O)cc1F C(=O)(CS(=O)c1ccc([N+](=O)[O-])cc1)NC1CCN(CC(=O)NC(C)C)C1 c1(C(=O)NCC(CNC(C2(c3cccc(C)c3)CC2)=O)F)nc[nH]c2ncnc1-2 c1(C(N2CCC(CC)C2CNC(=O)CC2CC3CCC2O3)=O)cc(F)ccc1C CCCCCCC(CC)C(=O)NC(C)C(C)NC(c1ccc(C2CC2)nc1O)=O N1(C(c2ccc(CC)s2)=O)CCCC(O)(CN(C)C(C2CCN(C)C2)=O)C1 c1(NC2CC(N(C)C(C3CC4CC4C3)=O)C2)cc(-n2ccnc2)ncn1 C(=O)(C(C#N)C(C)C)NC(C(=O)NCC(CC(C)C)OC)C CC1(C(=O)NC2COCC2NC(c2cn(C3CC3)cn2)=O)CCS(=O)(=O)CC1 C(=O)(CCCCCC(C)O)NCC(CNC(=O)C=Cc1ncc(C)[nH]1)OC C12(CNC(c3ccc(SC)o3)=O)CCCC1N(C(c1c(C)noc1C)=O)CCC2 c1(CC)ccc(C(=O)NCCCC(C)NC(c2ccnn2CCSC)=O)c(Cl)c1 C(CCS(=O)(=O)N1CC(F)CC1CC(=O)O)N(C)C C1(C(=O)NC(CC)C(F)(F)F)CC2CCCC2N1C(=O)C=C1CCCCC1 c1(C(=O)NC(CC)CN(C(=O)CCCNS(C)(=O)=O)C)cc(OC)nc(F)c1 CCC(C)C(O)C(C)C(=O)N1CCN(C)C(C(=O)NCc2cc(C)[nH]n2)C1 C(C)(CCC(=O)N(CC)CC)N1CCC(N(C(=O)COc2cccc(F)c2)C)C1 CC1CN(C(=O)C(c2ccccc2F)C2CC2)CCN1C(C1COC1)=O C1(NC(C2CC(OC)(OC)C2)=O)CCC(CC(=O)NCC(O)CC(C)C)CC1 N1(CCC(=O)NCCC(CNC(CN(CCC#C)C)=O)O)C(=O)CCC1=O c1(SCC)cnccc1C(=O)NC1CN(C(=O)C(C)C(c2ccccc2)SC)C1 N1(CCF)CC(C)OC(C)C1.c12ccc(cc1)n2C(c1cc(C(C)=O)[nH]n1)=O C1(C)(CC)CC(C(N2CCC(F)C(NC(=O)CCOCCOC)C2)=O)CCO1 c1(NC(=O)NCCC2(CO)CC2)cc(F)cc2c1OCCC2 C(=O)(CCCC(F)(F)C(F)(F)F)N(C)CC1(NC(C2Cc3nccn3C2)=O)CC1 C1(NC(c2cccc(CC)c2)=O)CCC2CN(C(=O)CC3CC3(C)C)CC2C1 Cn1c(C(=O)NC2CC3(C2)CN(C(C2CC(=O)NC(=O)N2)=O)C3)cc2sccc12 N1(C(C(C(C)C)N=[N+]=[N-])=O)CC2(C1)CN(C(c1cccc(O)n1)=O)CC(C)(C)O2 N1(C(COC(C)=O)=O)CC(CNC(C2CN3CCCC2C3)=O)C(F)(F)C1 C(=O)(C(C(=O)NC1(CN(C)C(c2ccccc2)=O)CC1)C(C)C)OCC C1(NC(=O)C=Cc2cnc[nH]2)CCN(C(c2ccn(C3CC3(F)F)n2)=O)C12CC2 c1(C(N2C(CNC(c3ccc(OC(C)(C)C)cc3)=O)CC2)=O)[nH]cc2c1CCC2 N1(C(C2N(C(C)C)CCC2)=O)CCOCC1CNC(c1ccc(N(C)C)cn1)=O CN1Cc2ccc(C(N3CCC(N(C(=O)CN4CC=CC4)C)C3)=O)cc2C1 N1(C(c2nc(CC)sc2N)=O)CCCC(CNC(c2cnn[nH]2)=O)CC1 CC1=NN(CCNC(C2CCOC(C(C)C)C2)=O)CCN1C CC1CCN(C(c2cccc(N)n2)=O)C(CNC(=O)CCC2CCC(=O)N2)C1 CC(C)(C)C(O)C(=O)N1CC=CC1CNC(=O)C=C(C1CC1)C1CC1 CC(C)(C)CCCC(=O)N1CC2CC2(CNC(c2cccnc2OC(F)F)=O)C1 N1(C(c2ncccc2F)=O)CCC2CC(C1)CN(C(C1CC=CCC1)=O)C2 C1(C(=O)NC2(C)CCN(C(CC3CC(C)OC3C)=O)CC2)CCC2(CCCO2)CC1 CC1CN(C(=O)C(Cc2ccoc2)NC(=O)C#CC(C)(C)C)C(C)CO1 c1(C(=O)NCC(C)(C(C)C)NC(C=C(C)Cl)=O)c(F)ccc(OC(F)F)c1F C12(C(=O)NCCSCCCCCO)CC(CN(C(=O)CCC3CCCCO3)C1)C2 CC(O)CCCCCC(=O)NC1(CNC(=O)CCn2cccnc2=O)CCC1 N1(C(C(CCCC)C(C)C)=O)CCC(C2CN(C(=O)C(O)c3ccsc3)C2)CC1 CC1C(=O)NC(C)CN1C(C1CN(C(c2ncsc2Br)=O)CC(F)(F)C1)=O c1(C(=O)NC2(C)CCN(C(C3(CC#C)CCC3)=O)CC2)c(C)ccc(C)c1O N1(C(CCCC(CC)(F)F)=O)CCC(CCC(c2ccccn2)=O)CC1 N1(C(c2c(CC)non2)=O)CCC(O)(CCNC(C2CCCC(O)C2)=O)CC1 C#Cc1cc(F)c(C(N2CCOC(CNC(C3(CC)CC3)=O)C2)=O)c(F)c1 C1(N(C)C)(OC)CCC(CN(C(F)(F)F)CC2CC(OC)C2)C1 C1(c2cn(C3CCN(C(c4ccc(SCC)s4)=O)C3)nn2)CCC(F)(F)CC1 C1(NC(CC2(CC)CC2)=O)CCCCC1CNC(C1(C)CC2CC2C1)=O CN1CCCC1CCC(N1CC(C(C)(C)O)(CNC(C2CNC(=O)N2)=O)C1)=O C(=O)(C(CC(F)F)NC(=O)Cc1cn(C)nc1C)NCC1C(C=C)OCC1 CCC(CC(F)(F)F)NC(c1ccccc1-c1ncnn1C)=O N1(C(C(C)C#N)=O)CC2CN(C(C34CCC(N(C)C)(CC3)CC4)=O)CC2C1 N1(C(C=NOC)=O)CCN(CCN(C)C(C2CCS(=O)(=O)N2)=O)CC1 c1(C(=O)NCC23CN(C(C4CC(=C)C4)=O)C(CO)(C2)C3)cc(OC)cc(OC)c1 C=CC(CC)CC(=O)N1CCC(NC(C2(CO)COC2)=O)C(CO)C1 N1(C(CC2N(C(CC(C)N(C)C)=O)CCC2)=O)CCC(F)(F)C(C)C1 N1(C(c2c(CCC)[nH]cc2)=O)CCCC(C2CC2NC(C2CCCS2)=O)C1 C1(NC(c2c(OC)scc2)=O)CC(NC(c2csc(O)n2)=O)C12CCOCC2 c1(C(N2C3CC(NC(=O)COCCF)CC2CC3)=O)ccc(F)c2occc12 CC1(C)C2CCC(C(=O)NCCOC3CCN(C(c4ccncc4)=O)CC3)C1C2 C1(F)(C(N2CC(CNC(C3(S(C)(=O)=O)CC3)=O)C2)=O)C2CCCCC12 c1(CC)ccnc(C(N2CCC(C(N3CCC(OCCO)CC3)=O)(OC)C2)=O)c1 CN1CC(O)CCC1C(N1CC(C(=O)N(CC(F)F)C2CC2)C(C)(C)C1)=O c1(C(=O)NC23CC(NC(c4c(CC)scn4)=O)(C2)C3)nnc(O)c2ccccc12 Cc1c(C2CC23CCC3)cccc1O.c1(C(CN)C)cccc(Br)c1 c1(C(N2C(CCCNC(c3c(C)csc3)=O)CCC2)=O)ccc2sc(C)nc2c1 c1(N(C)Cc2c(OC)c(Cl)ccc2)nc(=N)[nH]c(=NCCc2cncs2)[nH]1 C1(NC(c2c(C)ccc(C)c2)=O)CC2(CCC(NC(C3CCNC3=O)=O)CC2)C1 C(=O)(CC1CCc2ccccc21)NCC1(COC)CCN(C(C2CCCO2)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CN(C)C(c2ccccc2CO)=O)OCC1 Cc1nn(-c2cccc(F)c2)cc1C(=O)NC1CCC(c2nn[nH]n2)C1 N1(C(C(CCOC)N(C)C)=O)CC(CC(=O)NC2CC3CCCC3C2)C2(CC2)C1 C1(C(=O)NCCCCC(C)NC(c2cc(Cl)ns2)=O)CCc2nc[nH]c2C1 C1(CN(C)C(C2(C)CCCN2C)=O)CCN(C(C2CNC(=O)N2C)=O)CC1 N1(C(c2nc(COCC)sc2)=O)CCC(O)(NC(=O)COC(C)C)C1 c1(C(N2C(C)C(NC(=O)C=CC(=O)N(C)C)CC2)=O)ccc(Br)cc1F c1(C(N2CC3C(NC(c4ccc(OC)cc4Cl)=O)C3C2)=O)cc2c(nn1)CCC2 c1(C(N2CCC(C)(CNC(c3ccns3)=O)C2)=O)nc2ccccn2n1 C1(C(N2C(CC)C(C)(C)C2)=O)CCCCCN1C(=O)C(C)OCOC N1(C(c2cnc(OCC)s2)=O)CCN(C(=O)C(c2cncn2C)O)CC1C(F)F C1(CNC(C2CC(C)OC2)=O)COCCN(C(=O)C2=CCCOC2)C1 N1(C(Cc2cccc(C)c2)=O)CCC(C(=O)Nc2cccc(C)c2)C(O)C1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)C(C3CC3)SC)C(C)C2)=O)o1)NC CC1Oc2ccc(C(C)NCC(O)CN3CCCC3=O)cc2NC1=O c1(NC(C(C2CCOC2)NC(C(C)(C)n2cnnn2)=O)=O)cccc(N=[N+]=[N-])c1 N1(C(C2C(c3n(C)ncc3)OCC2)=O)CCCC(n2ccc(C(=O)O)n2)C1 Cn1cc(CN2CCOCC2CC(c2ccccn2)=O)c(O)n1 c1(CC(=O)NC2C(C)CCN(C(c3c[nH]c(Br)c3)=O)C2)ccc2nn[nH]c2c1 C1(C)(CNC(Cc2ccc(C)cc2C)=O)CN(C(=O)C(C)O)C(C)(C)C1 C1(C(=O)NCC2CC2CO)(CNC(=O)Cn2cc(Cl)cn2)CC12CCC2 N1(Cc2cccc(C(C)(C)C)c2)C(=O)CN(CC23CCCC2C3)C1=O Cc1ccncc1C=CC(=O)NCC1(C)CN(C(c2cn(C)[nH]c2=N)=O)CCO1 C(CC)(CCCC(=O)NC1(CCC)CCC1)NC(C1CNC(=O)C1)=O N1(c2ccnc(SC)n2)CC2CCCN(C(C3CC34CC4)=O)C2C1 c1(CC)csc(C(F)(F)C(=O)NC(C)CCNC(=O)CCn2ccnn2)n1 C1(COC)(CNC(=O)C(N2CCSCC2)C)CN(C(C2(F)CCC2)=O)C1 c1(NC2C(NC(c3cccc(Br)c3O)=O)C2)cccn2ncnc12 n1(CCC)c(CN2C3CN(C(=O)CCc4ccc(C(=O)O)cc4)CC23)nnc1C c1(-c2cn(C3CCN(C)CC3)nn2)cc(Br)ccc1Cl C1(C)(CNC(C(C)NC(C)=O)=O)CN(C(C2(CN(C)C)CC2)=O)CCO1 CC1CN(C(C2CC(=O)NC(=O)C2)=O)CCC1NC(=O)CN1CCCNC1=O CC(C)(F)C(C)(F)C(=O)N1CC(CNC(=O)CCc2nnc(C(F)F)o2)C1 C1(CNC(c2cn(CC=C)nc2)=O)CCCC(C(=O)NC2CCC(C(=O)OC)C2)C1 c1(OC)cncnc1C(=O)NC1CC(N(C)C(C2(Br)CC2C(C)=O)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NC(CC)CN(C)C(c1ncoc1C(C)C)=O C1(CC(=O)NC2(C)CN(C(c3nc(C(C)C)oc3)=O)C2)CCCNC1=O N1(C(C(CC=C)C)=O)CCCC(C(=O)NCCC2(C)N=N2)C1C C1(NC(C2(N(C(C)C)C)CC2)=O)CC(F)(CNC(CC(=O)Nc2nccs2)=O)C1 c1(C(=O)NCCC2CC(C(N(C3CC(CO)C3)C)=O)C2)cn(CCO)nn1 N1(C(c2c(CC)cc[nH]2)=O)CC2COCC2(C(=O)NCC(C)(F)C(C)(C)F)C1 Cc1ncc(C)c(NC(CNC(=O)C(=Cc2c[nH]cn2)F)C2CCC2)n1 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(c2c(C)cc(N)c(C)n2)=O)C(C)C1 N#Cc1ccc2cc(CNC3(CC#N)CCCOC3)[nH]c2c1 CCC(C)(C(=O)NCCN(C)C(c1nc(C(C)(C)C)cs1)C)OC C(C)(C)(CN=c1nc2c(c[nH]1)ncn2C)NC(C1=NOC(C)C1)=O c1(C(N(C(C)CN(C(=O)Cc2cccc(O)c2)C)C)=O)cnc2ccnn2c1 C(=O)(C1COc2ccc(F)cc21)NC(C(C)(C)C)CCNC(=O)OC(C)(C)C N1(C(c2cc(N(C)C)c(F)cc2)=O)CCC2(C1)CN(C(=O)C(F)CC(C)(C)C)C2 Cc1nc(N2CCC(C)CC2(C)C)nc2ccc(Br)cc12 C(=O)(C(C)C(=O)N1CCC(N(CCO)C(c2cccnc2S)=O)C1)OC CCC(C(=O)N(CCCC(N1CC2(CCC2)CC1C)=O)C)C(C)(C)CC C1(C2CC2)(NC(C(CC2CC2)NC(C2C3CN(C)CC32)=O)=O)CCOC1 N1(C(c2c(CC)cno2)=O)CCCC(CC2CCN(C(=O)C3=CCCC3)CC2)C1 CCC(CC)CC(c1nnnn1C1CCC1)NC1COC(CO)C1 CCC(CC(=O)N1CCN(C(=O)Cn2cncn2)C(CC(=O)NC)C1)CC(C)C C(C(=O)NC(CN(C)C)C(=O)NCC1(C)CC(C)=NO1)(C(C)C)SCC c1(OCC(N2CCC(CN(C(C3(CC)CCOC3)=O)C)C2)=O)cc(F)cc(Cl)c1 c1(C(=O)NC2CCCN(Cc3ccc(O)cc3O)C2)cc(O)c(O)c(O)c1 CCCC(CC1CCCCC1)C(=O)NCC(CC)NC(=O)CCOCC1CC1 c1(CNC(C(CC)CC)c2ccccc2)cc(Br)cc(Cl)c1O c1(CC(=O)NCCCN(C)CCO)ccc(C(=O)OC(C)(C)C)cc1.CC1C(=O)N1 C#CCC(O)C(=O)NC(CC1CCOCC1)C(=O)N(CCC)CC1CC1 N1(C(C2C(C)(C)CCN2C(=O)C2=NNC(=O)C2)=O)CCC2(CC(F)C2)C1 C1(C(N2CC(CC#C)OCC2)=O)CC2(CCN1C(=O)C(O)C1CCCC1)CC2 CCCCCCCC(=O)N1CCC(NC(=O)C(n2cc(Cl)cn2)C)C1CC N(C(=NCCNS(=O)(=O)C(F)F)N1CCC2(CC2)C1)C(C=C)C C1CCc2[nH]c(=NC3CCN4CCCCC34)[nH]c(=NCC3COCCO3)c2C1 CN1CCN(C(=O)C=C2CCC2)C(CNC(=O)C=Cc2ccccc2Cl)C1 C12CCN(CC1c1ccccc1)C(=O)N2.CC1OC2(CO)CC1C2 c1(C(C(=O)NCC(C)NC(CNC(C)=O)=O)(C)F)ccc(F)cc1 C1(C(N2C(CNC(C3(C)CC=CC3)=O)CCC2)=O)CCn2nccc2C1 N1(C(c2c(CC)ncs2)=O)CCCC12CCN(C(c1cnc(C)nc1C)=O)C2 C1(NC(C2OCC3COCCC23)=O)CCC2CCN(C(=O)Cc3ccon3)C1C2 c1(C(=O)NC2CC3(CN(C(C(COC)O)=O)C3)C2)cnc2cc(Cl)ccn12 Cc1sc(S(N)(=O)=O)cc1C(N1CC(N(C(=O)COC2CC2)C)C(C)(C)C1)=O C(=O)(CCCCCC(=O)OC)N1CCN(CCNC(CCC(=C)C)=O)CC1 CCN=c1[nH]cc(C(N2CC(C3(NC(C4CC5CCCC45)=O)CC3)C2)=O)s1 C(=O)(CCC(C)(C)NC(c1n[nH]c(=N)[nH]1)=O)N1CCC(C)(N(C)C)C1 c1(C(N(C(CNC(C(C)OCCC(C)C)=O)C)C)=O)ccc(C(=O)NC2CC2)cc1 c1(SCC(=O)NC2CCC(NC(c3n(CC#C)cnn3)=O)C2)ccccc1Cl C(C(C)N=c1nc(C#N)[nH]cc1C)N(C(C1(O)CCC(C)CC1)=O)C c1(C(=O)NCC2C(NC(Cc3scc(C)c3)=O)C2)c(Cl)ccc(O)c1Cl Cc1cc(C(=O)Nc2cc(N(C)C)ccc2F)nc(C)n1 C1(C(N2C(C)C(NC(=O)C=C3CCN(C)CC3)CCC2)=O)Cc2cccnc2C1 c1(C(C)NC(CC(COC(C)=O)(C)C)=O)cc(Cl)c(C)c(C)c1Cl c1(CNC(C2N(C(c3c(C)ocn3)=O)C3C(C2)C3)=O)n[nH]c2ccccc12 C1(CC=C)(NC(c2ccc(Cl)o2)=O)CC2CCC(C1)N2C(c1cc[nH]c1CC)=O C(N=C(NC(C)CC(C)C)N1CCOC(c2ccc(Cl)s2)C1)c1ccc(C)cn1 C=CCCC(C)NC(=O)C(CO)NC(=O)CC1CC1 N1(C(C(CC=C)(F)F)=O)CC2(C1)SCCC2NC(=O)CN(C(=O)COC)C c1(OC)cc(NC(=O)CC2CC(O)CN2C(c2sccc2C)=O)ccc1C C(CCCC(=O)N1CCC(C(=O)NCCN2CCOC2=O)C1)N(C)C(N)=O c1(OC)ccnc(C(N2CCN(C(c3cccnc3F)=O)CC2)=O)c1OC C12(C(=O)NC(CNC(c3ccn(C4CC4)n3)=O)C3CC3)CCCN1CCC2 N1(C(Cc2ccc(C)o2)=O)CC2CCN(C(c3cc(CC4CCC4)c[nH]3)=O)C2C1 c1(C(=O)NC(C2(CNC(c3cn(CC)nn3)=O)CC2)C)cccc(C)c1 Cn1c(CN2CCCC(NC(=O)CCCCO)C2)ccc1-c1ccccc1 N1(C(CC2(C#N)CCC2)=O)CCCC(NC(=O)C(c2ccccc2Cl)C2CC2)C1 C1(NC(=O)CC2CC2)CCCC12CN(C(=O)CCCn1ccnn1)C2 C(CC(C)(C)CC(=O)NC(CNC(c1cnn(CCF)c1)=O)CCOC)OC c1(OCC)ncc(C(=O)NC2(C)CC(NC(=O)CC3OCCO3)C2)cc1Cl C(=O)(C(F)CC(C)(C)NC(=O)C(C)C1CCC1)NC(CCC#C)C(=O)OC CCC(C)C(CN=c1nc2scnc2c(N(C)Cc2ccc(F)c(C)c2)[nH]1)OC Cn1cc(C(O)C(=O)NC23CC(CNC(c4ccoc4CC4CC4)=O)(C2)C3)cn1 N(C(=NCC1CCC1)N1CC2CC2C1)CC(c1ccc(F)cc1)NC(C)=O c1(C(=O)NC(CC=C)CNC(=O)CC(C)C(=O)OC)noc2cc(Br)ccc12 C1(C(N(CC(C)C)CC(=O)NCc2c[nH]c(C#N)c2)=O)CC12CCCCC2 c1(C(N2CCC(OCCNC(CC(CCC)C)=O)C2)=O)c([N+](=O)[O-])cnn1C N1(C(C2C(C)(C)C2)=O)CC2CC2(NC(c2ccccc2Oc2ccccn2)=O)C1 CC(CCN=c1nc(OC(F)F)cc[nH]1)NC(=O)CC(C)(C)C(=O)OC(C)(C)C C1(NC(CCCCOCC)=O)CCCCC12CCCN(C(=O)CSC(C)(C)C)C2 N1(C(C(CC)N2CCCC2=O)=O)CCC(O)(CN(C)C(C2CC(OC)C2)=O)C1 c1(N2CCC(NC(Cc3c(CC)cccn3)=O)C(O)C2)ccn2nccc2n1 Cc1nc(CNC(=O)C(=O)NCC2CC3(CC3)CO2)n(C)c1C C(=O)(CC(C)C(C)(C)C)OCCNC(=O)CO.CC1CNC(=O)CC1 n1(CC(=O)NC(C)CNC(C2CC3CC3C2)=O)c(=O)n(C)c2ccccc12 N1(C(c2c(SCC)nccn2)=O)CCC2(CCN(C(=O)C(C)C(C)CC)C2)C1 C1(CC=C)(C(=O)NC2(C)CCC(C)C2)CCCN1C(=O)C(=O)NC1CC1 c1(OC)ccc(C(=O)NCC2CCCN2Cc2cncc(OC)c2C)cc1C c1(C(=O)NC(CN(C(C(F)OC)=O)CC)C)oc(Br)cc1C C(=O)(C1=C(Cl)CCCC1)NC(CSCC)C(=O)NC(c1ccoc1)C CCCCC(CC)N=c1ccnc(NCC2CCCCNC2=O)[nH]1 C(C(COC)C(=O)NCc1cc(C(N2CCC2C(C)O)=O)cs1)OC C(C(=O)Nn1nnc(C)c1C)C1(CNC(C(CCC)C)=O)CCCC1 c1(NCC2N(OCC)CCCC2)nc(N2CCC(C)(CCO)CC2)cc(C)n1 CC(C(=O)NC(C)C(CO)NC(=O)Cc1ccc(CO)cc1)C(F)F c1(CC(=O)NC(C2CN(c3nccc(C#N)n3)C2)C)cccc2ccccc12 c1(OCC)cc(C)sc1C(=O)NCCCC(=O)NC1CC(CCSC2CC2)C1 N1(C(C(C)=C(C)C)=O)CC2(CCC(NC(C3CCc4nc[nH]c4C3)=O)CC2)C1 C(=O)(C(CO)NC(=O)CCn1cnnn1)NCC(C)C#N c1(CC)ccc(C(F)F)cc1F.c12ccc(cc1)NC(=O)C(=O)S2.C1CCCO1 C12(CNC(C3C(C)NC(=O)C3)=O)CC(CO)(CN1C(C1(C)CCCO1)=O)C2 Cc1cn2nc(C(=O)NCC3CN(C(C4CC4F)=O)C4(CCC4)C3)cc(C)c2n1 C(CCN(C(=O)CSCCC(F)(F)F)C)(C(C)C)NC(C1(CC)CC(C)(C)C1)=O C=CC(C)(CCOC)C(=O)N(C(CNC(c1cnn2ccn(C)c12)=O)C1CC1)C C1(C(N2CC(O)(C(C)NC(C(C)n3cccn3)=O)C2)=O)CC12CCCC2 N1(C(c2ccc(=NCC)[nH]c2)=O)CC2CCC(NC(=O)C(C)CF)CC2C1 C1(CNC(CCC#C)=O)CC2(CCN(C(c3cc[n+]([O-])cc3)=O)CC2)CO1 C(c1cncc(C)c1)=CC(=O)NC1C(CC)N(C(C2CC(C)C2)=O)CC1 C=C1CC2(C1)CC(C(N1CCC(C(C)NC(=O)C(C)(C)OCC)C1)=O)C2 C(=O)(C1CCOc2ccc(F)cc21)N1CCC(C)N(C(C2(CO)CCC2)=O)CC1 CC1CC(C(=O)NCC2(NC(C3CC(O)C3)=O)CCCCC2)CC(=O)N1 c1(C(N2C(CNC(C(CCCC)C)=O)C(C)CC2)=O)cc2c(F)ccc(F)c2s1 CC(C)S(=O)c1ccc(C(=O)NCCNC(=O)C(C(C)(C)C)OC(C)(C)C)cc1 N1(S(Cc2ccc(C(=O)OC)cc2)(=O)=O)Cc2cncnc2C1 N1(C(C2(O)CCN(C(c3ccc(CCCCC)cc3)=O)C2)=O)CCC(O)C(F)C1 C1(C(N(C(CNC(C=CC)=O)C2CC2)C)=O)CC2(CCC2OC)C1 C1(NC(=O)COc2cn[nH]c2)CCCCC1CNC(C1OCCO1)=O N1(C(c2ccc(OC)c(Br)c2)C(=O)NCCC2CC2)CCCc2ccccc21 Cc1ncc2n1CCC(C(=O)NCCC(C)NC(=O)CCS(C)=O)C2 C1(NC(CCOCC(C)C)=O)CC(CNC(=O)C2=NNC(=O)C2)C12CCC2 c1(C(=O)NCC=C2CCN(C(C3CC(C)(C)C3)=O)CC2)nc(O)nc(O)c1F N1(N2CCC2C=O)CC2CCC(C1)N2c1ccnc(-c2cccc(Cl)c2)n1.CC=O CCC(CCC(=O)N1CC(c2ccccc2)(NC(=O)CCCC(C)C)C1)OC C(=O)(CC(C)C(C)(C)NC(=O)C(C1CCC1)OC)NCC1N(C(CC)=O)CCC1 N1(Cc2ccc(OCC)nc2)CCC2(CCCN(C(=O)CCc3cnc[nH]3)C2)C1 C1(NC(C(C2CCCCC2)OC)=O)CCN(C(=O)CCF)C1C.c1(O)ccc(C)cc1 CC(C)(N=[N+]=[N-])C(=O)NC1C=CC(CNC(=O)OC(C)(C)C)C1 C1(C(=O)NCC2CC(CC)C2)CN(C(c2ccc(C#N)cn2)=O)CCC1C N1(CCNC(CC=CCC)=O)CCCN(C(c2[nH]ccc2C(C)=O)=O)CC1 C1(OC)COCCC1CC(=O)NCC(C)CNC(=O)CC=CCc1ccccc1 N1(C(c2[nH]ccc(=N)n2)=O)CC2(CCN(C(=O)Cn3ncc(Br)n3)C2)C1 c1(N2CC(CNC(c3ccc(F)s3)=O)OCCC2)ncnc2scnc12 N1(C(C2C(CC)C2)=O)CC2OCC(NC(=O)CN3CCC(F)CC3)C2C1 C(C(CC(C)C)C(=O)NCCCC(C)NC(=O)CCS(N)(=O)=O)OCC N1(C(C(=O)N(CC)CC2CC2)C2(c3ccccc3C)CC2)CCCC(CSC)C1 N1(C(CCC)=O)CC2CC1C2C(=O)Nc1cn(C)nc1Cc1cccc(Br)c1 Cc1cc(C(=O)NCC2CCCC(NC(=O)Cc3ccsn3)C2)cnn1 C1(CNC(CCNC(C)=O)=O)C(C)CCN1C(c1csc(C)n1)=O N1(C(C(C)CF)=O)CCC2C(CCN2C(=O)CCc2ccccc2O)C1 C1(O)(CCNC(C2CCCS2)=O)CCCN(C(C2SCCCS2)=O)C1 C(=O)(C(F)C(C)CNC(=O)CCC1CCOCC1)N(C)Cc1nc(C)[nH]n1 C(CC1=CCN(C(=O)CC(=O)OC(C)(C)C)CC1)NC(C1C(C)C1)=O.C(C)(C)C Cc1[nH]nc(C(=O)NCCCN(C)C(C2COCC2(C)C)=O)c1[N+](=O)[O-] N1(C(C)C)CC(C(=O)NCCC2(NC(C3CC4CCC3O4)=O)CCC2)CC1=O N1(C(C(C)SCCCC)=O)C2CCC(C2)C1CNC(c1cc(C)n(C)c1C)=O O(NC(=O)CC1CC1CNC(C)=O)CC#C.C1(=O)C=CC(C)N1 C1(C)(CNC(c2cc(CNC(CC=CCC)=O)no2)=O)NC(=O)NC1=O N1(C(CCc2scc(C)n2)=O)CCOCC(NC(C2(F)CC=CC2)=O)C1 c1(-c2ccc(OCOC)cc2)ccc2[nH]c(C(=O)NC3(C)CCCCC3)nc2c1 N1(CCNC(C2CN(C)C(=O)CC2)=O)CC2CCN(Cc3ccccn3)CC2C1 N1(C(c2cc(C#N)sc2)=O)CCC(O)C(NC(=O)CC2CC(=O)NC2=O)C1 C(=O)(CCC(CF)CF)Nc1ccc(C)c(NC(=O)CN(C)CCO)c1 O=C(CS(=O)(=O)C1CC1)NCC1CCC1NC(c1ncn2c1CCC2)=O N1(C(c2cc(CSC)c(F)cc2)=O)CCC2CCCN(C(=O)CC(C)(C)C)C2C1 C(=O)(C1=CCCSC1)N1CC(N(CC(=O)Nc2nccn2C)C)C2C1C2 C1(C(=O)NC2CC3(CN(C(C(CC)(C)O)=O)C3)OC2)C2Cc3cc(Cl)ccc3C12 CC(C)CCC(O)C(=O)N1CCCC(O)(CN(C(=O)CCc2ccccc2)C)C1 O(NC(=O)CCCC(C)NC(c1c(C)cccc1O)=O)CC.C=C1CC(C)C1 c1(C(=O)NCC(CC)(CC)NC(CC=CC=C)=O)cc(Cl)cc([N+](=O)[O-])c1O c1(C(=O)NCC(C)(CNC(=O)Cc2ccc(SC)cc2)OC)ncc(C)cc1F N1(C(C2C(CC)OCCC2)=O)CC2(CCCN(C(=O)C=Cc3csc(C)n3)C2)C1 c1(C(=O)NCCN(C(C2(CC(=O)OCC)CC2)=O)C)cn(C2COCC2=O)nn1 c1(CC)c(C(=O)N(C(C)CNC(C2(C)CCCCO2)=O)C)cccc1F CC1(NC(c2ccnn2C(C)(C)C)=O)CCN(c2ncc(Cl)cn2)C1 c1(CCC(=O)NC2CC(CCNC(C3CCCC3O)=O)C2)ccccn1 C=CCC(C(=O)N1CCC(CF)(NC(c2nncn2C)=O)C1)NC(C)=O O=C(CC1=NNC(=O)C1)NCCOC1CCN(C(C2CCCOCC2)=O)C1 N1(CCC(N2CCN(C(C(Br)=CC)=O)C3C2C3)=O)C(=O)NC(C)(C)C1=O c1(NC(CONC(=O)NCC(C)N(C)C)=O)cccc(Cl)c1F C(=O)(CCCCC(C)C)NCC1CC(F)(CNC(c2cccc(OCC)c2)=O)C1 c1(C(=O)NC2CCN(C(c3c(=N)[nH]cnc3)=O)C2C2CC2)cnc2nccn2c1 N1(CC(=O)N(C)CCN2C(CC)COCC2)CCN(C)CC(C)C1 CC1(C)C(NC(=O)COc2ccc(Br)cc2F)C2CCOC12 N1(C(c2c(OC)nsc2)=O)CCC(C2(NC(=O)Cc3cccc(OC)c3)CC2)C1 N1(C(CCC(C)OC)=O)CCC(CNC(c2ccc(C(N)=O)o2)=O)C1(C)C CCCC(C(=O)N1CCC(CNC(=O)C(c2ccc(Cl)c(Cl)c2)O)CC1)C(C)C c1(CC)cscc1C(=O)NC1CC(C)(NC(=O)C(C)OCC2CCCCO2)C1 CC1CC(NC(c2cccnn2)=O)CN1C(=O)CCCc1ccccn1 N1(C(C(COCC)NC(c2ccc(Cl)o2)=O)=O)CCOC(CF)C1 C(C)(C)CCCCCC(=O)N1CC=CC1CNC(c1cc2sccc2n1C)=O c1(C(N2CCC(CNC(CC(C)n3cccc3)=O)C2)=O)cnn(C)c1F N1(C(CCC2CN(C(C3N(C(C)=O)CCC3)=O)C2)=O)CC(C)NC(=O)C12CC2 Cc1cccc(C)c1-n1cc(C(C)N(C)C(c2ccc(F)cc2)=O)nn1 CCCCCCCCC(=O)N1CC(c2cn(C(C)C(=O)OC)nn2)(C(=O)OC)C1 C(C(C(=O)NC1CCCC1SC)C(C)(C)C)NC(c1cc(OCC)n[nH]1)=O N#Cc1ccc(NC(C2CCN2Cc2ccc(N3CCCC3=O)cc2)=O)s1 N1(C(C2N(C)CC(O)C2)=O)CCN(C(=O)Cc2ccccc2O)C(C2CCC2)C1 c1(OC)cccc(Cn2c(-c3n[nH]c(C)c3C)nc(CCc3ccccc3)n2)c1 CC1COc2c(C(N3CCC(NC(=O)CC4CCOC4)C(C)C3)=O)cccc21 c1(OC)cc2c(s1)CCN(C1CC3CC1N(C(c1cccc4ncnn14)=O)C3)C2 N1(C(C(C)(C)OC)=O)CCN(C(=O)C(C)(C)C(N)=O)CC12CCC2 C1(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)(NC(CCC=C(C)C)=O)CC1 N1(C(C2(SC)CCC2)=O)CC2CCCC(N(C)C(C3CCCCC3C)=O)C2C1 Cc1cc(CNC(=O)CCC2CN(C(=O)CCCC3CCC3)CC2C)ccn1 c1(C(N(C2CN(C(=O)C(C)(C)CF)CC2(C)C)C)=O)c(Cl)nc2cc(Cl)ccn12 C(=O)(C1COc2ccc(Cl)cc21)N1CCCCC(NC(C2=CC(C)(C)C2)=O)C1 c1(C(=O)NC2C(CNC(C3C(C)C3C)=O)C2)c(F)ccc2occc12 C(=O)(CC1COc2cc(O)ccc21)NC1CCN(C(c2c(C)c(N)cnc2)=O)C1 C(CC(O)CC(=O)NC1CCCC1NC(C1(C)CCOC1)=O)SC c1(C(=O)NC2CN(C(C3C(OCC)C3C)=O)C(CO)C2)ccc(C)cc1O c1(SC)ccc(C=CC(N2CCC(C)(NC(=O)CC3CC3)C2)=O)s1 C(=O)(C1COc2ccccc21)N1CC(NC(=O)CC2CCCC2)CC12CCC2 N1(CCC)CCCN(C(=O)C(COCC)NC(=O)C2=CCCCO2)CC1 C1(C(=O)NC(C)CCNC(=O)C(C2CCCCCC2)C)CC(=O)NC1(C)C c1(C(c2nnnn2C2CC2)NCC2(OCC=C)CC2)ncoc1C(F)F c1(C(C(C)C)NC(COCCOC)=O)ccccc1OC.C12CC(C)(C1)NC2=O N1(C(C=COCC)=O)CCC2OCCN(C(c3cccc(N)c3)=O)C2C1 N1(C(c2cc(C(=O)OC)nn2C)=O)CCN(C(c2cnccn2)=O)CC1C Cc1cncc(C(N2CCC(O)(CNC(C3CCC3C(C)(C)C)=O)C2)=O)n1 C1(SC)CN(C(=O)C(C)(C)n2cccn2)CC1NC(=O)C(C)CC1CCCC1 c1(C(=O)NC(CC=CC)C(=O)NCCCCC)cc2ccccn2n1 C(=O)(C1(CC)CCc2ccccc21)NCCN(C(=O)C#CC1CCCCO1)CC C(C)(C(=O)N1CCC(C(C)C(=O)NCCCC(=O)NO)CC1)(C(C)C)NC(C)=O c1(C(=O)NC(CNC(C2C(OC)(OC)CC2)=O)C(C)(C)C)cc(Cl)ccc1C C#Cc1cc(NC(=O)Nc2ccc(CC3CN(C)C(C)(C)C3)cc2)cc(F)c1 C1(NC(c2cccc(C)c2)=O)CC2CC1CN2C(C1CC1c1sccc1C)=O Cn1cc(C(=O)Nc2cccc(NC(=O)Cc3nc[nH]n3)c2)c(C(F)(F)F)n1 CC1CCC(C(c2nnnn2C)NCc2sccc2Br)CC1 C=C1CCC1(C(=O)NCc1cnn(Cc2ccccc2)c1)C(=O)OC C(=O)(CC(CN(C)C1CC1)CC)N1C(CNC(CC2(C(=C)F)CCC2)=O)CC1 C(CC(O)C(F)(F)F)NC(C1(OC)CCN(C(Cc2cc(CC)no2)=O)C1)=O C(CNC(=O)CCn1cnnn1)(CC(C)C)NC(c1c(CC(C)C)onc1)=O N#Cc1ccc(NC(c2ccccc2NCC2CCCS2)=O)c2cccnc12 C12(C(=O)NC3(C(C)(F)F)CC3)COCC1CN(C(=O)CCc1ccoc1)C2 c1(C(=O)NC23C(CN(C(CCN(C(C(C)C)=O)C)=O)C2)C3)ccc(F)nc1F C=CC(C)(CCOC)C(=O)NCC1(OC)CN(C(=O)CC2CC(C(=O)OC)C2)C1 CC(C)(C(=O)NC1CCC1NC(=O)C(F)(F)C(F)F)C1=CCS(=O)(=O)CC1 c1(NC(=O)CCc2cncs2)cc(F)ccc1C(F)F.C12CC(C1)CNC2=O S(=O)(=O)(C1CCN(C(=O)CC2(C(=O)O)CCCC2)CC1)N(C(C)C)C C(CCC(C)(C)NC(=O)COCCCN=[N+]=[N-])NC(C(c1ccn(C)c1)C)=O c1(-c2n(C)ccn2)cccc(NC(=O)CCc2ccnn2C)c1 C(C(CNC(=O)COc1ccc(Cl)cn1)C(F)(F)F)NC(C(CC)OCC)=O Cc1n[nH]c(=NCC2CC(CNC(c3cc(C4CCCN4C)[nH]n3)=O)CO2)s1 C=CCN=C(NCCc1cccc(C#N)c1)NCC(F)(F)Cc1ccccc1 c1(C(=O)OCC)ccc2c(c1)NC(=O)CN(C(=O)NC(c1ccoc1)C)C2 CCC(C(=O)N(CCCNC(c1ccc(-c2ccco2)o1)=O)C)N(CC)CC c1(CC(C)C(=O)NCCCNC(C2(c3ccco3)CC2)=O)ccccc1F CC(CC(F)F)C(=O)N1CCCC1CNC(C1CCCN1C(=O)CC(C)C)=O N1(C(CCN(C(C)=O)C)=O)CC(NC(c2n[nH]c(C3CC3)c2Br)=O)C(C)C1 c1(C(N(CCCNC(c2n(C(C)C)ccc2)=O)C)=O)cnc(Br)c(N)c1 N1(C(C(=CC2CCCC2)C)=O)CC2CC2(NC(=O)Cc2ccc(Cl)cn2)C1 Cc1ccc(C(=O)NCCCCN(C(=O)CCC2CC2(F)F)C)c([N+](=O)[O-])c1 C1(C2CC2)(NC(c2coc(C3CC3)n2)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 c1(C(=O)NCCC(C)NC(C(C)OCC)=O)cccn(C)c1=O C(=O)(C(C(C)(C)C)C(C)(C)OC(C)(C)C)N1CC(F)(C(=O)OC(C)(C)C)C1 C(c1ccsc1)=CC(=O)NC(Cc1cccnc1)CO C1(COCC)CCN(C(C2C3CN(c4ncccn4)CC23)=O)CC1 C1(CNC(CSCC(=O)OC)=O)CCC(NC(=O)C(c2cccc(F)c2)O)CC1 c1(OC)ccccc1C(CNC(C)=O)NC(c1sc(-c2ccccc2)nc1C)=O O=C(NNc1ncnc2cc(Cl)ccc12)c1coc2c(F)cccc12 C1(CC#C)(C(N2CCC(NC(C34CC(CO3)C4)=O)CC2)=O)CC=CCC1 Cc1c(Cl)nc[nH]c1=NCC1(O)CCCN(C(=O)C(C)NC(=O)OC(C)C)C1 c1(OCCOC)ccc(C(=O)NCC(C(C)C)NC(=O)Cc2ccns2)cc1 c1(OCC(=O)NCC(CC)(C)NC(=O)CC2(C)CC2)ccccc1Br c1(C(=O)NC2(CF)CN(C(C(C)(C)c3ccno3)=O)C2)ccnc(S)c1 N1(C(CC)C(=O)NCC(C)CNC(C2CCC2)=O)CCC(N(C)C)CC1 C1(OC)(CNC(c2ccc(C(F)F)o2)=O)CCN(C(=O)C2CC2)C1 c1(CN(C=O)Cc2c(F)cccc2Cl)ccc(F)c(C(F)(F)F)c1 N1(C(C(=O)Cc2cccs2)=O)CCCC12CCN(C(c1sccc1OC(F)F)=O)C2 C1(CCNC(C(C2CCOCC2)OCC)=O)CSCCN1C(c1cc(Cl)cs1)=O n1(CC)cc(C(N2CCC(C)C2CNC(=O)C(C)(O)C2CC2)=O)c(C2CC2)n1 N1(C(CC(C)C)=O)CCC(C2CC2)(CNC(C2CC3(C2)CC(O)C3)=O)C1 c1(C(N2C(C)C(NC(c3csc(C4CC4)n3)=O)CC2)=O)cnc2ncccc2c1 C1(CC(=O)NCCC(N2C(CC(C)C)COC2)=O)CCN(C)CC1 C1(C(=O)OCc2scc(Br)c2Br)(COC)CCCCO1 c1(C(N2CCC(NC(C34CCCN3CCC4)=O)C(O)C2)=O)cncc2sccc12 C#CCC(C)(C)C(=O)NCC1(F)CCC(NC(c2cc(C3(O)COC3)on2)=O)C1 c1(NC(C(CCF)NC(COCC)=O)=O)cn(C)c(=O)nc1O N1(C(C(C)=C2CCC2)=O)CCC2(C1)CN(C(=O)C(C)C1CCC1)C2 C(S(=O)(=O)c1ccccc1)c1c(CNC(=O)NC(C)C(F)F)cccc1 CCCC(C)(CCC)C(=O)NCC1(F)CCN(C(C2(C)CC2(F)F)=O)C1 Cc1cccc2oc(N3CCC(CF)(NC(=O)CSc4cnn(C)c4)C3)nc12 C#CCC(C)(C(=O)NC1CC(CO)C2CC12)NC(C1CC(CCC)C1)=O c1(C(=O)NC2C(C)CCN(C(C(CC)N(C)C)=O)C2)c(C)ccc([N+](=O)[O-])c1C N1(C(C2CCN(CC(C)C)C2)=O)C2CCC(C2)C1C(N1CCOCC1C)=O C#CCCCCCC(=O)NC(CO)C(=O)NC(CC=C)C1CC1 Cc1cc(C(c2ccccc2F)NCC2CCCCCC2)ccc1OC(F)(F)F C1(C(N(CC(C)N(C(=O)Cn2ccnn2)C)C)=O)CCc2nc(O)nc(O)c2C1 N1(C(C(COC)(C)C)=O)CC2CS(=O)(=O)CC2(NC(c2cccn2C2CC2)=O)C1 CC(C)CC(C)(O)C(=O)N1CC(CNC(C23CCCC(C2)OC3)=O)C(C)(C)C1 C(c1ccc(O)cc1)=CC(N1CC(CCNC(C2CC23CC3(F)F)=O)C1)=O C(=O)(CC(C)C(F)(F)F)NCC1(C(=O)NCc2c(C)noc2CC)CC(=C)C1 C#Cc1ccc(C(=O)NC(C2CCN(C(c3cncnc3C(C)C)=O)C2)C)o1 Cc1cccn(CC(=O)OCc2cn(CCC3CCCCC3)nn2)c1=O CC1CC(NC(=O)NC(Cc2ccccc2Cl)CO)CC(C)S1(=O)=O C1(CC=C)(NC(=O)C(C)CF)CCN(C(c2cc(NC(C)=O)cnc2C)=O)CC1 CC1(NC(c2nncn2C2CC2)=O)CCCN(C(c2c(F)cccc2F)=O)C1 c1(C(N(C2CCCN(C(C(C(CC)C)OC)=O)C2)C)=O)cnc2ccccc2c1 Cc1cccc(C(N2CCC(NC(=O)CC3CC4CCC3O4)C(C)C2)=O)c1F N1(C(CSCC#C)=O)C2CCC1CC(CNC(C1COCCN1C=O)=O)C2 c1(OC)c(Cl)ccnc1C1CC(=O)NC(=O)N1.c1(SC(C)(C)C)ccncc1 C1(N(C(C(CC#C)O)=O)C)CC2CCC(C1)N2C(=O)C(F)C(CC)CC CCCC(C(=O)NC1CCCC1NC(c1nc(C)oc1C)=O)NC(C)=O N1(C(CNC(=O)OC)=O)CCN(C(c2cnc(Cl)c(F)c2)=O)C(CO)C1 Cc1ccc(C(=O)NCC(C)N(C)C(c2cc(-c3ccco3)c[nH]2)=O)s1 c1(CC(N2CC(C)C(NC(c3cncc(Br)c3)=O)C2)=O)ccc2nonc2c1 C1(NC(COCC#C)=O)CCCC(CC(=O)NC(c2cnn(C)c2)C(N)=O)C1 c1(C(N2CC(C(=O)NC3(C(O)CO)CC3)OCC2)=O)cc2cnccc2[nH]1 N1(C(C(C)OCCC=C)=O)CCC2(CCN(C(c3nc(O)sc3C)=O)CC2)C1 C12(CNC(C=CC)=O)CC(NC(=O)CCc3ccsc3Cl)(C1)C1(CCC1)O2 C1(C(C)O)CCN(C(=O)Nc2ccc(-n3cccn3)cc2)CC1 C1(CNC(C(c2ccccc2)N(C)C(N2CCCC2)=O)=O)CC=CCC1 c1(NC(CCC)=O)cc(CNC(=O)C(O)CC(C)C)c(F)cc1F Cc1ccc(OCC(=O)NC2(CNC(c3c(C)cnn3C)=O)CCOCC2)cc1 CC1CN(C(c2nc(Br)ccc2F)=O)CCCN1C(=O)C=Cc1ccccc1Br c1(OCC#C)ccc(C(=O)NCC2CC(F)CN2C(=O)CC2CSC2)cc1 c1(CS(=O)(=O)Nc2ccc(CC(=O)NC)cc2)ccc(Cl)cc1[N+](=O)[O-] CC1CN(C(=O)C=Cc2ccncn2)CCC1CNC(C1(O)CCOCC1)=O N1(C(CCCCSC)=O)CCC(NC(c2cc(Cl)c(C)cn2)=O)C(F)C1 O=C1CCC(CC(N2CCCC(O)(CNC(C3(O)CCC3)=O)C2)=O)C(=O)N1 CC1CN(C(c2cc(C3CC3)on2)=O)CC2(CCN(C(=O)CCS(N)(=O)=O)C2)O1 C1(NC(C=C(CCC)CCC)=O)CCN(C(=O)C(C(C)C)OCC)CCC1CO Cn1nc(C(=O)NCC2CC(NC(c3sccc3F)=O)C2)c2c1CCSC2 C1(CNC(CCCN(C(CN2CCC(C)C2)=O)C)=O)CCC(F)(F)C1 c1(C(N2CC(C(N3CCC3)=O)(CC)C2)=O)cnc[nH]c1=N.c1(C2C(O)C2)ccccn1.C c1(-c2nc(C=O)sc2)cc(F)ccc1F.CC1(C2=CC=C2)CCCN1CC(C1CC2OCCC12)=O C1(NC(C2C(C)C2)=O)CC12CCN(C(c1cccc(C(F)F)c1)=O)CC2 N1(C(CSCC)=O)CCC2CN(C(=O)CN(S(=O)(=O)c3ccccc3)C)C2C1 CCCCC(C)C(=O)NCC1CC(C)N(C(=O)CSCc2csc(=N)[nH]2)C1 c1(OC)ccncc1C(c1nnnn1CC1CCCO1)NC1CC(n2cccn2)C1 N1(C(C=CCOC)=O)CC(C)CCC1C(=O)Nc1ccccc1.C12CC1OC2 N1(C(c2ccc(C)cc2)=O)CCCC(CCNC(C2(C)CC2C)=O)CC1 C1(NC(c2c(CC)nco2)=O)CC2CCC(C1)N2C(C1CC1CC)=O c1(C(=O)NC2(C)CN(C(c3n(COC)ncc3)=O)C2)cc(C)cc(Br)c1 c1(NC(c2cncc(-c3cc(C)c(C)nc3)n2)=O)cnn2cc(Br)ccc12 c1(C(=O)NCC2C(NC(c3c(OCC)nccc3)=O)C2)ccc(P(C)(C)=O)cn1 c1(CCC)c(C(=O)N(C)CC2COCCN2C(=O)C(C)OCC)cnn1C CC(CC(F)(F)F)C(=O)NC1CN(C(c2ccc(NC=O)cc2)=O)CC(F)(F)C1 c1(OC(C)C)ccccc1C(=O)NC1CC(N(C)C(C2(O)CCOC2)=O)C1 C1(CCC)(NC(=O)CCC(=O)NCC)CCN(C(c2cc(C(N)=O)no2)=O)C1 C(=O)(C(O)CC(N)=O)N(C)CC1OCCN(C(c2cc(CC)c(C)s2)=O)C1 c1(NC2CC(NC(=O)CC3=CCCC3)C2)ncnc2[nH]cc(I)c12 n12nc(-c3ccco3)nc1C(O)C2.c1(CC(c2ccccc2)O)ccccc1F C1(CNC(c2ccnnc2O)=O)CCCC(NC(C2CC(n3cnnc3)C2)=O)C1 C1(CC)CC(C(=O)NCC(C)N(C)C2CC2)CCN1C(C1C2CCC(F)C12)=O N1(C(C(COC)OC)=O)CCCN(CCCCNC(=O)Cc2ncc(C)s2)CC1 c1(C(N2CC(CCNC(c3cncnc3)=O)(OC)C2)=O)cccc(CCC#N)c1 c1(C(CC(=O)NCC(c2ccsc2)O)N(C(=O)COC(=O)C2CC2)C)ccccc1 Cc1cn2c(=O)c(C(N3CC(F)(C(N4CCC(=O)C(C)C4)=O)C3)=O)cnc2s1 c1(N2CCC(NC(C=C(C(=O)OC(C)(C)C)F)=O)C2)ncccc1F C1(NC(Cc2nc(C)sc2)=O)CC(NC(c2cnoc2C)=O)CC1O N1(C(COC2CC(C#N)C2)=O)CCCC(NC(c2nncs2)=O)CC1 Cc1coc(C)c1C(=O)N(C1CCN(C(=O)C(C)(F)F)C1)C C1(C(CNC(C(COCC)C)=O)(C)C)CCN(C(=O)C=CC2CCOC2)CC1 C1(C(=O)NC(C#C)CC(C)C)C(C)OCCN1C(=O)C#CC(C)(C)O N1(C(c2nc(CC)oc2)=O)CCCC(C)(C)C1CNC(=O)CNc1nccs1 c1(C(=O)NCC2CCC(C(=O)NCc3cccc(Cl)c3)O2)cc(F)ccc1O C1(C(N(CC(CC)(O)CC)C)=O)CC2(CC(NC(C3CC(C(C)C)=NO3)=O)C2)C1 c1(C(=O)NCC2(NC(CC(c3cccc(F)c3)C)=O)CCOC2)c[nH]n(C)c1=O C(C)(C)(CCCNC(=O)Cn1cnnn1)NC(CN(C(COC)=O)C)=O C(=O)(CCC[N+](=O)[O-])NC1(CC=C)CN(C(C2CCC(=O)N(C(C)C)C2)=O)C1 CN1CCC(C(N2CCC2CC(C)(C)C)=O)C1=O C1(C)(NC(C(CCOC)C)=O)CCN(c2ncc(F)cn2)CC1 N1(CC)CCCN(C(=O)CC2(CNC(c3cc(C#N)oc3C)=O)CC2)CC1 N1(C(CCOC)=O)CCCC1C1CCCCN1C(C1CC(C(F)F)(OC)C1)=O c1(OCC)cc(COC)ccc1NC(=O)Nc1nccc(CC#N)n1 n1(CC(=O)NCC23N(c4nccc(CC(=O)OC)n4)CC(C2)C3)ccc(O)nc1=O N1(C(C2(C)CC2C(F)(F)F)=O)C2CCC1CC(NC(C1(CF)CCC1)=O)C2 C(C)(C(=O)Nn1nnc2c1CCCC2)N(C(=O)C(C#N)C(C)(C)C)C(CC)=O c1(C(N(c2cc(OC)ncn2)CC2CNCCO2)=O)c(F)ccc(C)c1Br c1(C(=O)NCC2(CNC(Cc3ncc(COC)[nH]3)=O)CCC2)c(Cl)cncc1Cl N1(C(CN2CCN(S(CCCNC)(=O)=O)CC2)=O)CC(F)(CO)CC12CCC2 C12(F)COCCN(C1)C(=O)CO2.C(C(O)COC)NC(COCC)=O C(=O)(C1=CS(=O)CCC1)N1CCCC(C)(NC(=O)COC2CCCC2)C1 C(c1ccc(Cl)cc1)=C.C(=O)(CC)N(CC(C)NC(=O)CCOCC1CCCO1)C Cc1ccc(C(N2CCC(OCCNC(=O)CN3C(=O)CNC3=O)C2)=O)c(N)n1 c1(CC(N2CCCC(n3cc(C4(OC)CCC4)nn3)C2)=O)ccc2c(c1)OCO2 C(=O)(C1=CC2(CN(C(C3CC3F)=O)C2)OC1)N1CC(C)(C)C(C(N)=O)C1 c1(C(C)OCC)nc(-c2coc(Cl)n2)n(Cc2cccs2)n1 c1(C(=O)NC(C(C)C)CCNC(=O)Cc2cnnn2C)cccc2oc(=N)[nH]c12 C1(CNC(c2nc(C(N)=O)sc2)=O)CN(C(=O)C2CC2)CC(c2ccccc2)O1 N1(C(=O)OC(C)(C)C)CC2(CCOCC2)CC1CC(=O)Nc1cccc(CO)n1 C(=O)(CCS(=O)(=O)N(C)C)N(CC(CC)NC(=O)Cc1nocc1C)C C1(c2nc(COCC)nn2-c2ccn(C)n2)CCCCC1(C)C C1(NC(c2ccc(C(C)C)o2)=O)CN(C(=O)C(C)NS(C)(=O)=O)CC1C C(=O)(CCCCCC(C)(C)C)NCCCN(C(C1CC2(C(C(=O)OC)C2)C1)=O)C c1(NC(N=c2c(C)cn(C(C)C)[nH]2)=O)c[nH]c2ccccc2c1=O c1(C(N2CCC(CC=C)(C(=O)NC3CC(C(C)(C)C)C3)C2)=O)cc2occc2[nH]1 c1(CC)nc(C)c(C(=O)NC2(C(=O)NCCCCC3CC3C)CCCC2C)o1 N12CC3(C1)CN(C3)CC2.c1(NC(CN(CC)CC)=O)cn(C(C)C)cn1 C1(C2CC2)(NC(C2OCCN(CC)C2)=O)CCN(C(=O)Cc2cnn(C)c2)C1 c1(C(C(=O)NCCOC)N(C)CCOCC2CCCCC2)cc(Br)ccc1F C(C)(CC(C)NC(c1cnc(CCCC)s1)=O)NC(C1(C#C)CC1)=O c1(C(=O)NCC(C2CC2)NC(C(c2ccc(C)cc2)C)=O)c(F)ccc(C)c1F C1(NC(C(CC)CC(F)F)=O)CCC2(CC1)CN(C(=O)CC(C)(C)CC)C2 Cc1cc(C(N2COC(C)(C)C2)=O)ccc1-n1cc(CO)nn1 N12CCCn3nc(cc3C1)C(=O)Nc1cc(F)ccc1C2.N1(CC)CC(O)C1 N1(CCCC(=O)NCCN(CCC)C(C2CC=CC2)=O)Cc2ccccc2C1=O N1(C(c2nn(C)c(C#N)c2)=O)CC(C2CN(C(=O)CN3CC4CC4C3)C2)C1 c1(OC)ccc(C2CN(C(c3nn(C(C)C)cc3Br)=O)CCO2)cc1 c1(OC)ccc2c(c1)CC(C(N1CCCN(C)CCC1)=O)O2 c1(C(N(CC)Cc2ccnn2C)=O)ccc(C(=O)NCCC(=O)OC)nc1 C(CS(=O)(=O)C1CCOCC1)NC(C1(C(F)(F)F)CCCC1)=O c1(C(N2CC(NC(c3c(C)[nH]nc3Cl)=O)C3C2C3)=O)c[nH]c2c(F)cccc12 c1(CN(C)C)ccoc1C(=O)N(C(CNC(=O)C(F)n1ccnc1)C1CC1)C C(C1=NOC2CN(C(=O)COc3ccccc3)CC12)NC(c1ccnc(C)n1)=O C1(NC(C=CC(CC)=CC)=O)C2CC3CN(C(=O)CC4CCC(=O)N4)C1C3C2 c1(C(=O)NC2CCN(C(Cc3c(C)c[nH]n3)=O)C2)cc(O)ccc1O C(=O)(C1CCCc2n[nH]cc21)N1CC(C2(NC(c3cccc(SC)c3)=O)CC2)C1 CCC(COC)C(=O)NC(C)C(CO)NC(=O)CNC(=O)C=Cc1ccccc1 C1(N(C(COCCNC(C2(C(=O)OCC=C)CC2)=O)=O)C)CC12CCCCC2 C1(C(N2C(C(C)(C)NC(c3cnc(O)o3)=O)CCC2)=O)CC2C=CC1C2 C1(C(N2CCN(c3ccccc3)CC2)=O)CC2CCC1N(C(=O)C(Cl)(Cl)Cl)C2 c1(C(N2C(C)CC(NC(c3nc(CCC)sc3)=O)C2)=O)cnn2ncccc12 C1(CNC(C=CCC2(NC(Cc3ccn(C)n3)=O)CCC2)=O)CCNC(=O)C1 C(=O)(C1=C(F)CN(C(C2CCC2C)=O)CC1)NC(c1cnsc1)C C(=O)(C(F)(F)C(F)(F)F)NC1CN(C(C=CC(C2CCOCC2)=O)=O)CC1O Cc1cc(C(=O)NC2CCCC2C(=O)NC(C2CCCOC2)(C)C)n(C)n1 CC(C)C(O)C(F)(F)C(=O)NC1CC2CC1CC2C(N1CC(C)C(N=[N+]=[N-])C1)=O Cc1ccc2nc(C(=O)NCC=CCNC(=O)CC3CCC(C)C3)ccc2c1 c1(OC)cn(C)c(C(=O)NCCC(C)NC(=O)C(C)=C2CC2)cc1=O C(C(CC(=O)N1CCC1CC(C)(C)C)NC(=O)CCc1ccncc1)OC N1(CC(COc2cccc(OCCC)c2)O)CCSC2(CCCC2)C1 C1(NC(C2C(CCC(C)C)CCC2)=O)CCOC(C(C)(C)C)C1 N1(C(C2CC(C)C2)=O)CC(NC(=O)Cc2cc(Cl)cc(Cl)c2)C(F)(F)C1 N1(C(Cc2ccc(C)o2)=O)CCC(C2CCN(C(=O)CCCS(N)(=O)=O)CC2)C1 CC(c1ccccc1C)=CC(N1CCC1CNC(C1CSCCS1)=O)=O CCCCC(F)C(=O)NC(CN(C)C)C(=O)N(C(CC)CC)CC N1(C(c2ccc(I)c(F)c2)=O)CCC2C1CCCN2C(c1c(Cl)cccc1I)=O C#Cc1ccc(C(=O)NCC2CN(C(=O)CCN(C)CC)CCO2)s1 N1(C(=O)NCc2c(C)ccc(CN(C)CC3CCCO3)c2)CCC(=O)N(C)CC1 CCC(CCC(=O)N1CCC(C(=O)N(C)OCC(F)(F)F)C12CC2)OC CON(CCC(=O)NCCc1cccnc1)C(=O)c1cc(Cl)cs1 C1(C#CC(=O)N2CC(NC(=O)CC3CCC(O)C3)CC(C)(C)C2)(CC)COC1 C1(NC(c2nc(C)sc2C)=O)CC2CC(C1)N(C(=O)CC1CCCCC1(C)C)C2 C(CN=c1[nH]c2c(c(=NC(C)Cc3cnn(C)c3)[nH]1)CCC2)NC(C)C C1(C2(O)CCC2)(CNC(C2C(C(C)NC(C3CC4(CSC4)C3)=O)C2)=O)CC1 N#Cc1ccc(CNCC2COCC2Sc2ccc(Cl)cc2)nc1 C1(COC)(CNC(c2cnc(SC)s2)=O)CN(C(=O)C(O)Cc2ccccc2)C1 CC1CN(C(=O)CCNC(C2CCC2)=O)CC(C)C1C(=O)NCc1ccnn1C c1(C(=O)NCCCN(C(CCc2ccc(C)o2)=O)C)ncc(C2CC2)cc1F C1(CNC(c2n(C)nnc2-c2ccccc2)=O)CC2C(O)CC2O1 C(CCO)(C(=O)NCC1(NC(=O)CCCOc2ccccc2Cl)CC1)N(C)C c1(OCC(N2CC3(N)CCCC3(F)C2)C)cccc2c1OC(C)(C)C2 C1(CCNC(=O)Cn2ccnn2)(NC(=O)C=Cc2ccsc2)CCOCC1 CN1Cc2c(-c3csc(C(N4CCC5(CCOC5)C4)=O)c3)cccc2C1=O C1(C(N2CC(F)(CNC(Cc3c(C)con3)=O)C2)=O)Nc2ccccc2C1(C)C C(=O)(C(F)C(CC)CC)NC(C(=O)NC1(C#C)CCOC1)(C)C1CCC1 CC(C)(C(=O)NC1CCC1CNC(c1ccsc1C(F)F)=O)CS(C)(=O)=O CC1CC(c2ccc(Br)cc2)CN1C(=O)CCN1C(=O)CCC1=O C#CC(C)(C)C(=O)NC(C1CCCN1C(=O)C(C)=CC1CC1)C C#Cc1cccc(C(=O)NC2CCC(N(C(=O)CNS(=O)(=O)NC)C)C2)c1Cl CC1C(NC(c2cc(O)nc(O)c2)=O)CCCN1C(c1cc(CO)[nH]n1)=O c1(-c2cn(C(C(N3CCC(OC(C)C)C3C)=O)C)nn2)cc(F)c(F)cc1F c1(CNC(=O)C(N2CCC(F)C(O)C2)C2CC2)ccc2c(c1)CCC2 c1(SC)ccc(C(=O)NC2(C)CN(C(C3CCS3(=O)=O)=O)C2)cc1 c1(C(C)N(CC(C2CCCNC2)=O)C)nccc(-c2ccccc2)n1 N12CCN(CC1)NC2=O.c1(CC2CCCO2)nnnn1CC1(CO)COC1 N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CC(NC(C2CCC(C)(C)CC2)=O)C(C)(C)C1 N1(C(COCCCOC)=O)CCN(CC(C)NC(=O)CC2CC(C)=NO2)CC1 c1(CC)nc(=NC(CCN(C(=O)C(O)Cc2ccccc2)C)C(C)C)s[nH]1 c1(C(=O)NCC2(C)CCN(C(C(C3CCC3)OCC)=O)C2)cccc2nonc12 c1(C(=O)Nc2cccc(-c3ncn(C)n3)c2)ccc2nc(Br)nn2c1 c1(N2CC(CC)OC(CC)C2)nc(=N)[nH]c(=NCCc2cc(C3CC3)no2)[nH]1 c1(CC)ccc(NC(=O)NCc2ccccc2F)cc1C(F)(F)F N1(C(CS(CC)=O)=O)CCC2CN(C(c3ccc(O)cc3C(F)F)=O)CC2C1 C(=O)(C1=NNC(=O)CC1)N1C(C2CN(C(CC#C)=O)C2)CCCC1 CC(C)C1=CCC(NC(C2CCN(C(=O)CC3CC(=O)NC3=O)CC(O)C2)=O)CC1 CC1CCOCC1C(=O)NCC=CCNC(=O)CCOc1cccc(C(N)=O)c1 C1(C(=O)NCC2(C(=O)NCC3CSC3)CC2)CC1C1CCC1 Cc1ccc(C(C)C)cc1C(=O)NC(C)Cc1ccc(OC(F)F)c(C(F)(F)F)c1 N1(C(C(C)N(C)C(=O)OC(C)(C)C)=O)CCN2C(=O)CCCC2C1 c1(C(=O)NCCc2nc(O)n[nH]2)csc2cc(Br)ccc12 S(=O)(=O)(c1cnc(NC2COc3ccccc32)c(Cl)c1)NCC1(CC)CCCO1 c1(N2CC3CN(C(Cc4cccc(CC)c4)=O)C3C2)nc(C)nc2ccsc12 N1(C(C(CC)N(C)C)=O)CCC(C)C(NC(c2ccc(SC)o2)=O)C1 Cc1cc2ncc(C(=O)NCCC3CC(NC(=O)Cc4nocc4C)C3)cn2n1 C(c1ccc(F)cc1F)=CC(=O)N(C(CNC(C=Cc1ccc(C)o1)=O)C)C N1(C(CNC(CC)=O)=O)C2CCCC1CN(C(=O)Cc1ccc(S(C)=O)cc1)C2 c1(C(N2CC(NC(C3N(CCC)CCC3)=O)C2)=O)cc(C(F)(F)F)ccc1C c1(CCOC(CC(CCC)C)=O)ccc(N2CCCC2)c([N+](=O)[O-])c1 C(=O)(CC1=CSC2=NCCN12)NCC1OCCN(C(C2(C)CC(C)(C)C2)=O)C1 c1(C(=O)NC(CC=C)CC(=O)NCC(CC)CCCC)ccc2nncn2c1 CC1CCC(CNC(=O)Cn2cccn2)N(C(=O)CN(C)C(c2ccoc2)=O)C1 Cn1ccc2c(NC(=O)CCC3CCCN3Cc3cc(I)ccc3O)ncnc12 CC1C(C(=O)NC2CC(CF)C2)CCN1C(c1cccc(O)c1)=O N1(C(=O)Nc2ccc(S3(=O)=NCCC3)cc2)CCc2ccc(O)cc2C1 N1(C(CCOCC#C)=O)CC2CCN(C(C3CC4C=CC3C43CC3)=O)C2C1 CC1CN(C(c2ccnc(N(C)C)c2)=O)CCCN1C(=O)CN(CCO)CCO CCCCC(CNC(c1cccc(N(C)C)c1)=O)NC(C1CCC(=O)NC1C)=O c1(SC)ccc(-c2cn(C(C)C)nn2)cc1.c12ccc(cc1)C(=O)NC1CCC21 c1(N2CCC3(CCN(C(c4ncccc4Br)=O)C3)C2)ncnc2cccc(F)c12 C(=O)(C(C)NC(C)(C)CC)NC(CN(C(C=CCC)=O)CC)C C1(N(C)C)CCCN(C(=O)C(N2CC(O)CC2C2CCC2)=O)C1 Cc1nc(NCC(O)CNC(=O)C(C)Cc2ccc(O)c(O)c2)cc(O)n1 c1(C(N(CCCNC(c2cn(CCC)nc2C)=O)CC)=O)ccc(OC)cc1F CCC(CC)C(C(=O)N1CC(NC(=O)C2=NNC(=O)C2)C1)N1CCOCC1 CC1=C(C(=O)NC(C)(C)CC(N2CCCOCC2C)=O)COCC1 C1(NC(C(C)S(C)(=O)=O)=O)CCC2CN(C(C3CCC4(C3)N=N4)=O)CC2C1 C1(C(N2CCC3(CN(C(=O)Cc4csc(Br)n4)C3)C2)=O)CCC2(CC1)OCCO2 N1(C(c2occ(CC)n2)C(=O)NC2CC(F)(F)C2)CCCN(S(N)(=O)=O)CC1 C=CC(O)C(=O)NCCCC1(NC(=O)CC2CC(CC(C)(C)C)C2)CC1 C(=O)(CCC[N+](=O)[O-])NC(CC(C)NC(C1(COC)CC1(F)F)=O)C C(=O)(C(COC)NC(c1cc(C(C)=O)c[nH]1)=O)N(CCCCC)C C1(NC(C2N(C)CCC2)=O)CCCC12CCN(C(c1cn(C)nc1Cl)=O)CC2 N1(C(CCC(C)N(C)C)=O)CC2CC1CN(C(c1cnn3c1CCC3)=O)C2 C1(C(C)C)(CNC(c2cn(C)cn2)=O)CCN(Cc2ccc(Cl)nc2)C1 c1(C(=O)NC2CN(C(C(C)NC(C)(C)C)=O)C(C)(C)C2)coc2c(Cl)cccc12 C1(C(=O)Nc2cc(F)c(Cl)cc2F)CCC2(CN(Cc3ccc(I)cc3)C2)O1 c1(C(=O)NC2CC(C)(CNC(c3cc(CO)on3)=O)C2)cn2cccc(Cl)c2n1 n1(CCC(N2CCCC(N(C(=O)Cn3cccn3)CCO)C2)=O)cccnc1=O C=C(Cl)CC(C(=O)NCCc1cc(C)no1)NC(c1cc(=N)[nH][nH]1)=O CC1CN(C(=O)CC2CCSCC2)CCN1C(=O)C=Cc1cocn1 C(CC(C(C)(C)O)N(C1N(C(CCC)=O)CCC1)C1CC1)NC(c1ccco1)=O C=CCC(CC(C)C)C(=O)NCC1CN(C(c2cocn2)=O)CCC1C(F)(F)F c1(CNC(C(C)NC=O)=O)ccc2c(c1)CN(C(=O)C1Cc3ccccc31)C2 C1(C)(C(=O)NC(C(=O)NC(C#C)CC)Cc2cc[nH]n2)C(C)(C)C1(C)C N1(C(C2C(OC)CC2)=O)CCC(C)(CNC(=O)C=C2CCCCC2)C1 c1(-n2cc(CC(C(=O)NCCc3n(C)ncc3)O)nn2)ccccc1Cl CC1(NC(c2cc(C(N)=O)co2)=O)CC(NC(C2CSC2)=O)C1 C1(CNC(C(Cc2ccoc2)NC(c2cnns2)=O)=O)CCC(O)CC1 CC(CN(C)C)CC(=O)NCCCN(C(c1ccc(CCO)cc1)=O)C1CC1 CC1(C)CN(C(=O)C2=CCSC2)CC1CNC(c1ccc(N(C)C)nc1)=O c1(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC=CCC2)cc(C(N)=O)co1 N1(C(C(c2cccc(F)c2)(C)OC)=O)CCCCC1C1CCOC1 C1(C(=O)NCCCC(F)(F)F)(COC)C=CCN1C(=O)CSC Cc1nc(C)c(CNC(=O)C(C2CC=CCC2)NC(c2cn(C(C)C)cn2)=O)s1 CC1(NC(N2CCC2CO)=O)CC1(Cl)Cl c1(OC)ccc2c(c1)CCC2C(=O)NC(C)CCC#N N1(C(C(C)S(C)(=O)=O)=O)CCN(C(=O)CC2(C3CC3)CC2)CC12CCC2 C12CN(CCC1c1ccccc1)C2.c1(SC)cc(C(=O)OC(C)(C)C)sc1Cl C=CCC(C)(C)CC(=O)N1CCC(C(C)NC(c2c(C)cccc2C)=O)C1 C1(C(=O)NC(CNC(c2c(C)nncc2)=O)(C)C(C)C)CCC2(CC1)CC2 c1(C(=O)NC(C2CCCCC2)CNC(=O)CCn2cccn2)cccc(CO)n1 C1(C(=O)OC)CCOC1C(=O)NCC1(NC(=O)CN(C)S(N)(=O)=O)CC1 CC(C)(CCC(=O)NC1CCCC(C(=O)NCc2cccc(O)n2)CC1)[N+](=O)[O-] c1(C(=O)NC2C(C)CCN(C(c3ns[nH]c3=O)=O)C2)ccc2c(c1)NCCC2=O C(=O)(C(C)(C)C(C)NC(C1CC2(C1)CC2(F)F)=O)NCC#CCOC Cc1c[nH]cc(C(=O)N(C2CCCN(C(=O)C(N3CCSCC3)C)CC2)C)c1=O N1(C(C2CC(O)(CC#C)C2)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])s3)=O)C2C1 C(CCC(C)(C)NC(=O)CCn1cccn1)NC(C1C(C)CCS1)=O C1(CNC(c2cnc(C(C)OC)s2)=O)CN(C(=O)CC=CC(C)(C)C)CC1(C)C C1(C(=O)NCCN2CCOCC2)CC2CCC(C1)N2C(=O)C(c1ccccc1)F C1(c2c(C34CCOC(C3)OCCO4)n(C)c(=O)[nH]2)N(C)N=CC=CO1 C#Cc1cc(C(=O)NC(C)C(=O)NCC)ccc1C.C1(C)(CO)C(=O)N1 CCCS(=O)(=O)C(C)C(=O)N1CC2(CCCN(C(C3CCOC(=O)N3C)=O)C2)C1 C1(NC(C=CC(=O)OCC)=O)CC12CC(NC(c1ccnnc1)=O)C2.C1CCCC1 N1(C(C(C(=O)OC)C)=O)CCCC2(CCN(C(c3cccc(Cl)c3C)=O)C2)C1 O(NC(=O)C(F)C1CCN(C(c2csc(O)n2)=O)C1)C(CC)C O(NC(=O)C=CC(C)SC)CC(=O)N(C1COC(=O)N1)CCN1CCCC1.CO CN(C)C(=S)NCC(=O)N(C1CC(C(N)=O)C1)C CCN(OC)C(=O)CNC(=O)C(C)(C)C1CCCN1C(c1ccoc1Cl)=O C1(NC(C2N(C)CCOC2)=O)CN(C(c2[nH]nnc2C2CC2)=O)CCC12CCC2 c1(NC(CCC)C2CC2)cc(C)c(S(=O)(=O)N2CCC2CF)cn1 CC(CN(C)C)C(=O)NCCCCC1(NC(c2c[nH]c(Br)c2)=O)CC1 C1(C(=O)NC(c2nc[nH]n2)CO)(COC)CN(C(c2c[nH]nc2C)=O)C1 C(CO)(CCCCNC(c1cnn(CC)c1)=O)NC(C=CCCC)=O O=S1(=O)CCCC2CC(NCc3nc(C4CCOCC4)n[nH]3)C12 c1(C(=O)NCCN(C)C(c2c[nH]nc2C2CCCO2)=O)cccc(F)c1Cl c1(C(=O)NC(C2CCN(C(C3CC(O)C3)=O)C2)C)cc2c(cc1Cl)OCO2 Cc1ccc(C(N2CCC(O)C(NC(c3c(C)csc3Cl)=O)C2)=O)cc1Cl C(C(=O)NC1CCCCC1NC(=O)CCCC1CCC1)(C(C)C)OCC(C)C N=c1[nH]c2ccc(C(=O)NCC3CC(NC(=O)CCOCC(F)F)C3)cc2s1 CC(C)(CC(=O)NC(C(=O)O)C1CC1C(=O)O)n1cc(-c2cccc(Cl)c2)nn1 CCCCCCC(F)C(=O)NC1CC(CNC(=O)CC=CC(C)(C)C)CC1O C1(CNC(=O)COCCF)CC12CCN(C(C1CCC=CCCC1)=O)CC2 C(=O)(C(C)C(C)(F)F)NCC(C)N(C(C=CC(C)=O)=O)C C(=O)(CCC(C)(F)F)NC(C(N1CC(C)OCC1)=O)C1(O)CCC1 c1(C(C(=O)NC(C)(CNC(=O)C=CC(F)(F)F)C2CC2)F)ccccc1 C1(C#CC(=O)NC(C2CCN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)C)(CC)CC1 c1(OCC)cc(C(=O)NCCC2CCCN2C(=O)C(C)(F)F)ccc1OC(F)F N1(C(c2nccc(CC)c2)=O)CCCCC(NC(=O)COc2cccc(C)c2)C1 N1(C(COC)=O)CCCCC(N(C(=O)C(Cc2ccccc2)OC(C)C)C)C1 CC1=CCN(C(=O)CCC2CC2(F)F)CC1.C12(CC1)C(=O)NC2C C=CC1(c2cn(CC3CCN(C)C3)nn2)COCCN1C(c1cnn[nH]1)=O c1(CC)ccc(C(=O)NCC(C(C)C)NC(=O)CCn2ccccc2=O)nc1 C1(NC(C=CCOC)=O)CCC12CCN(C(=O)CC(C)n1ccnc1)CC2 C1(C(N(C2CC(NC(C3(C)CC(C(=O)OC)C3)=O)C2)C)=O)CC2(CCC2)CO1 N12CCC(CC1)CN(CCC)C2=O.C(C)(C)(C)NC(=O)CC C12(CNC(C(c3ccc(Cl)s3)C)=O)CCC(CC1)N(C(=O)CC1CCC(=O)N1)C2 CN1CCC(C(=O)NCCCSC(F)F)(NC(=O)CC2CC(=O)NC2=O)C1 c1(-n2ncc(C(=O)NC(C)C(C)NC(c3cncn3C)=O)c2)cccc(F)c1 N1(C(c2ncc(NC)nc2)=O)CC2CCC(C1)N2C(=O)Cn1nccc1N N1(C(c2n(CC=C)ccn2)=O)CC(NC(c2nncs2)=O)CC1(CC)CC c1(OC)ccc(C(F)(F)F)cc1NC(C1CCCN1C(=O)C(F)CC1CC1)=O N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CCC(C1)N2C(=O)C=CC1(C)COC1 C12(C(C)C)CC(C(=O)NCCN(C(=O)C(c3ccc(Cl)s3)C)C3CC3)(C1)C2 c1(C(N(C2CN(C(c3coc(CO)c3)=O)CC2O)C)=O)ccc(OC(F)F)cc1 Cc1nc(C2CC2)oc1C(=O)NC1(C)CCN(C(=O)C(C)CO)C1 Cc1cc(C(=O)NC2CN(C(c3ccccc3)=O)CC2(F)F)cc(C)c1 C(CCCCC)(C(=O)NCCC)NC(C(C)N(C1(COC)CC(=C)C1)C)=O c1(C(=O)NCC2(O)CN(C(C3(F)C(C)C3)=O)C2)cccc2sncc12 C1(NC(CCCOCC=C)=O)CCN(C(=O)C=Cc2c[nH]nc2C)C12CC2 c1(C(=O)NC(C)(C)CNC(=O)Cn2nccn2)cccc(Oc2ccccc2)c1 N1(C(c2cn(CCCC)nn2)=O)CCN(C(C2CCCCN2C)=O)CC1CF C(=O)(C(O)P(C)(C)=O)N1C(CNC(CCC(c2cc(C)sc2C)=O)=O)CCC1 C(=O)(C(C)CC(C)(C)C)NC(C(=O)N(CC(C)C#N)C)(C)C C1(C(N(C2CCN(C(c3ccc(CO)s3)=O)C2)CC)=O)CCC=CCCC1 C1(C(=O)NC(C)CC2(O)CCC2)CN(C(C2C(C#N)C2(C)C)=O)CC12CC2 C1(CNC(C(CSC)C)=O)CN(C(c2ccc3sncc3c2)=O)C2(CCC2)C1 C1(NC(CCC(=C)Br)=O)CC(F)CN(C(=O)C=CC(=O)OCC)C1 N1(CC(=O)NC2CCCC2NC(=O)C2=CCOC2)CCCCCC1=O C1(NC(C(C)(C)C(N)=O)=O)CCC2CC1CN2C(c1cnn2ccccc12)=O C1(NC(C(CC=CC)CC)=O)CC2CCC1CN2C(=O)Cc1cc(F)ccc1C N1(C(c2cn(CC(F)(F)F)cn2)=O)CC(NC(C2(Br)CC2)=O)CC(O)C1 CN1C(=O)CCC1C(N1CCC(F)(C(=O)NC2CC2N)C1)=O C1(CN(C(=O)Cc2nccs2)C)CN(C(=O)CC2CC3CC3C2)CCO1 Cc1cc(N)c(C(N2CCCC(CNC(C3CCCC(F)(F)C3)=O)C2)=O)cc1C N1(C(CC(CCC)CC)=O)CC2CC(C)N(C(=O)COC(F)(F)F)C2C1 C1(CCNC(C2C(C(C)NC(c3cc(C(F)F)no3)=O)C2)=O)CCN(C)C1 Cc1cc(C(N2CC3C(CNC(=O)COc4ccn(C)n4)C3C2)=O)cc(C)c1O N1(C(c2cc(C)nc(O)n2)=O)CCC2(CC(NC(=O)CSCC(C)C)CO2)C1 C1(C(=O)NC2(C(=O)NCC(C(CC)C)C)CCOCC2)CCCCC1(C)C c1(NCCN(CC(=O)N(CC)CC)C2CC2)ccc(=O)n(CCC(C)(C)C)c1 CC(CCCCNC(C1(CF)CCOCC1)=O)NC(c1ccc(C(F)F)o1)=O CCCCC(C(=O)NCC1CC1)NC(=O)Nc1ccccc1C1CC1 C(C)(CC(C)NC(c1occc1Br)=O)NC(CSCCC(C)C)=O C1(NC(N2CC(CCC)N(C(C)C)CC2)=O)CCCC2(CCCC2)C1 N1(C(CC(C(C)C)C)=O)CC2CN(C(c3c[nH]nc3C(C)(C)C)=O)CC2(C)C1 CCC(C)C(C)CNC(C1(SC)CN(C(c2ccc(C(F)(F)F)nn2)=O)C1)=O c1(C(=O)NCC(CC(=O)NCC2(O)CCCC2)OC)cc(O)ccc1C N1(C(C(C)SC)=O)CCN(C(c2cc(C(F)F)cs2)=O)CC(O)C1 C1(NC(c2cc(CC)n(C)n2)=O)CCN(C(=O)Cc2cccnc2OC)CC1F C=CCCC(F)(F)C(=O)N1CC2(CCC2NC(c2coc(-c3ccsc3)c2)=O)C1 N1(C(CCNC(=O)C=CCl)=O)CCCC12CCCN(C(=O)CC(F)F)C2 CCCCC(O)C(=O)NCC(F)CNC(c1csc(CC(F)(F)F)n1)=O N12CCC(CC1)OCC2=O.N1(C(C(=O)NCC(C)OCCOC)=O)CCC(C)C1 c1ccccc1OC(F)F.c1(C2(C)CN2)nnnn1CNC(=O)OC.C1CC1.OCC C(=O)(CCCC(=O)N1CCC(C(=O)N(C)CCc2ccncc2)C(C)C1)OCC Cc1cccc(C(=O)NCC(C)(C(C)C)NC(=O)CSC2CCOC2=O)c1F CCCCC(C)CCC(=O)NC(CNC(=O)CNC(c1ccoc1)=O)CCC CCCCC(O)C(C)C(=O)NCC1CC(CCC(N2CCC23CCCSC3)=O)C1 c1(N2CC(C)SC(C)C2)ccc(S(=O)(=O)NC2(n3cc(C#N)cn3)CC2)cc1Cl Cc1c(C(N2CCN(C(=O)Cc3cc(F)cc(Cl)c3)CC2CF)=O)cncc1Cl CCCCC(C)(F)C(=O)NCC(C)CN(C(=O)C(N1CCCCCC1)C)C C1(COC)CN(C(=NCCc2cn(C)nn2)NCSC)CCO1 Cc1cc(C(=O)NCC2CC2CNC(c2cccc(C(F)F)c2)=O)ccc1Br Cc1ccc(C(=O)NC2CCC2NC(c2nccn2C(C)C)=O)c(Cl)c1 N1(C(c2occ(C)c2)=O)C2CCC1C(C(=O)NCCSCC(=O)N(C)C)C2 C(C(C)CN=c1nc(CCSC)[nH]s1)NC(c1c(COC)cccc1)=O N1(C(C2CC(CCC)C2)=O)CCC(NC(c2ncsc2C)=O)C(F)C1 C1(NC(C2N(C(C(CCOC)C)=O)C(C)C2)=O)CCCN(C)CC1 Cc1nc(C(=O)NC2CCCC2NC(=O)CC(C)(C)C)nn1C Cn1nc([N+](=O)[O-])cc1C(=O)NCC1(NC(=O)Cc2ccc(Cl)c(F)c2)CC1 c1(C(=O)NC2CC(F)(CNC(C=CC=CC)=O)C2)ccc2cccnn12 CC(C)CC(C)(CNC(=O)C=Cc1cccc(Cl)c1)NC(=O)CCS(C)=O C1(C)(C(N2CC(C)C(F)C2)=O)CCCN(C(=O)CN2CCNC(=O)C2)C1 Cn1ncc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2CC=CC2)cc1=O C1(O)(CNC(c2c(OC)cccn2)=O)CCCN(C(=O)COC2CCCC2)C1 c1(CC(=O)NCc2c[nH]nc2C(=O)Nc2ccc(CO)cc2)cc(O)cc(F)c1 CC(C)CC(C(=O)NCC#CCNC(=O)CCc1ccccc1Br)C(C)C N1(c2cccc(C(COC(=O)CCc3ccoc3)=O)c2)CCC(=O)NC1=O Cc1ccc(C)n1CC(=O)NC(C)CN(C)C(C1(O)CC(C)(C)C1)=O C1(OC)CC(CC(N2CC(O)(CN(C)C(c3ccc(C)s3)=O)C2)=O)C1(C)C C(=O)(C1=CCC(C)CC1)N1CCCC(NC(c2c(Br)ncc(C)c2)=O)C1 Cc1cccc2c1CCOC2C(=O)N1CCC(NC(c2nnn(C)c2C)=O)C1C Cn1nc(C(=O)NCCCNC(C2(C)CC2F)=O)c(C(F)(F)F)c1Cl C1(C(=O)NCCN(C(C(C=CC)O)=O)C(C)C)CCCC12CC2 c1(C(C)NC(=O)C(C)(C)CN(C)C(C2CCN(C)C2=O)=O)cc(F)ccc1F O=C(C1COc2ccc(F)cc21)N1CCOC(Cn2cc(-c3nc[nH]n3)nn2)C1 C1(O)(CNC(CC(C)C2CC2)=O)CCCN(C(C2(C)CCC(=O)N2)=O)CC1 C(=O)(CCS(=O)(=O)N(C)C)NCC12C(CN(C(C(C(C)C)OCC)=O)C1)C2 C(=O)(CC(C)C(C)(C)NC(=O)CCCN(C)C(=O)OC)N(CC#C)CCO C(=O)(C1CCc2cc(F)ccc21)N(C1CCN(C(CS(CC#C)(=O)=O)=O)C1)C c1(C(=O)NC(CC)CN(C)C(c2cncc(O)c2Cl)=O)cc(C2CC2)ccc1Cl C1(C(C)(C)C)C(NC(=O)CC2COC(=O)N2)CCN1C(=O)CSC(F)(F)F C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(c1ccc3nsnc3c1)=O)C2 c1(CSC)cc(C(=O)NC2COCC2NC(c2cnccc2C)=O)sc1C C1(OC)CN(C(C2(O)CC2)=O)CC1C(N1CCN(CC(N)=O)CC1)=O C1(CC(=O)N(C(C)COCC)C)CC(O)C1(C)C.C1C(=O)N1CC#C Cc1ccc(C(N2CC(F)CC2C(=O)Nc2c[nH]nc2C#N)=O)cc1F N1(C(c2ccc(N(C)C)cn2)=O)CCCCC(NC(=O)CCC2CCC2)C1 N1(C(c2c(OC)csc2)=O)C2CCC1CC(CNC(=O)CCc1cc(C)no1)C2 N(C(=NCCCN1CCCC1=O)NCC(C(F)(F)F)C(F)(F)F)C(c1cccs1)C N1(c2cc(OCC)ncn2)CCC2CN(Cc3ccc(CC(=O)OC)cc3)CCC12 C(=O)(CCCNC(=O)C(C)(C)C)N(C1CC(NC(=O)C(F)OC(F)(F)F)C1)C c1(CC)cc(C(N2CC(NC(C3CCN3C3CCCC3)=O)C(O)C2)=O)cc(N)c1 N1(C(c2cc(C)ncn2)=O)CCC2(CCCN(C(=O)CN3CCCC3C)C2)C1 C=CCC(CC)C(=O)NC(COC)CC(=O)N(CC(O)C(F)(F)F)C N1(C(c2cc(C)c(C)o2)=O)CCOC2(C1)CN(C(c1sc(C(C)C)nc1C)=O)C2 Cc1noc(NC(=O)OC(C)(C)C)c1C(=O)NN(C)CCSC1CCSC1 c1(NCc2ccn(CC(N3CC4C(C(=O)OC)(C4)C3)=O)n2)cc(C)cc(C)c1 C#Cc1ccc(C(N2CCC(O)(CN(C(=O)C(F)=CC)C)C2)=O)c(F)c1Cl Cc1cc(O)ccc1C(=O)Nc1ccc(-n2ncnc2C)cc1 c1(CC(=O)NC2C3CN(C(c4cn(CC)nc4)=O)C(C3)C2)nn(C)cc1[N+](=O)[O-] C1(C#N)(NC(C(C2CCCN(C(c3ccc(C)cn3)=O)C2)C)=O)CCOCC1 c1(CC)cc[nH]c1C(=O)NCC1(C(=O)N(C23CC(C2)C3)C)CCCO1 c1(C2C(C(N(C)CN)=O)C2)ccccc1NS(=O)(=O)Cc1ccccc1 c1(C(=O)NCC2CN(C(C(CC)SC)=O)CC2C)cccc2c1OCC2 N1(C(CCNC(=O)CO)=O)CCC(C(=O)NC2COCOC2)CC1 N(C1CCOc2cc(F)cc(F)c21)C(C(C)Oc1ccc(F)cc1C(F)(F)F)=O c1(C(N2CC(C)N(c3nc(Cl)ncc3Br)CC2)=O)cnn2ncccc12 c1(C(=O)NC2CC3CCC2N(CC2(C(F)(F)F)CC2)C3)ccc2ccccc2n1 c1(C(CNC(N2C(C3C(O)CCC(C)C3)CCC2)=O)=O)ccc2c(c1)OCCO2 c1(CC(=O)NCC(C2CC2)NC(CSCC)=O)coc2cc3ccccc3cc12 c1(C(=O)NCC(CN(C)C(c2cccnc2)=O)(C)C)cc(=O)cc(Cl)[nH]1 S(=O)(=O)(c1cccc(F)c1)N(CC(=O)NCC1N(C(CCOC(C)=O)=O)CC1)C CC1=NN(C)C(=O)C1CC(N1CCC(NC(C2(C(C)C)CC2)=O)C1)=O C=CC1CN(C(=O)CCCNC(=O)CCn2cccc2)CCO1 CC1(NC(C(=O)NCc2nnsc2-c2ccccc2)=O)CCCNC1 Cc1cc(C(=O)NC(C)C(CO)NC(C2(n3cnnn3)CC2)=O)co1 C1(C(=O)NCC2C(CNC(C3(C(F)(F)F)CC(=C)C3)=O)C2)CC2CC1C1CC21 c12ccc(cc1)C(=O)NC2.c1(C(=O)OCC=C)cn(CC(C2(CC)CCC2)=O)nn1 C(CCN=c1nc2sccc2c(NC(C)CN2CCCC2)[nH]1)(C(C)C)OCC Cc1cccc2c1OC(C(=O)N(C)CCOCCCNC(c1sccc1F)=O)C2 Cc1cc(O)c(CNC2CC(NC(c3cc(=O)cco3)=O)C2)cc1Cl Cc1ccc2c(c1)CCN2C(c1cc(F)ccc1N)=O C=CCCCCCCCCCCNC(=O)NCC1(C)CCOCC1 c1(C2C(c3cn(C)nc3)N(C(c3cc[nH]n3)=O)CC2)ccn2nccc2n1 Cc1cc(C(N2CC(N(C(=O)Cc3cncs3)C)C(C)(C)C2)=O)nnc1O c1(C(N(C)CCNC(C2CC(n3ccnc3)C2)=O)=O)cc([N+](=O)[O-])sn1 N1(C(C(COCc2ccccc2)OC)=O)CCC(NC(=O)C2=CSCS2)C1(C)C C(=O)(C1CCc2cccnc21)NC1CCC2(CCN(C(C(C)O)=O)C2)C1 N1(C(C2CCN(C(CCCOCCC)=O)C2C)=O)Cc2n[nH]cc2C1CO N1(CCC(=O)N(CCCNC(=O)CCc2scnc2C)CCC)CCC(C)CC1 N1(C(c2c(C)c(Cl)cnc2)=O)CCC(NC(=O)CCC(C)C)C(CO)CC1 N#Cc1ccc(Cl)c(NC(N2CCCC(C(=O)Nc3ncccn3)C2)=O)c1 C(N(O)C(=O)C1COc2ccccc21)c1cn(CCCCCC(N)=O)nn1 C(=O)(C1CCc2snnc21)NC(CNC(C(CC(CC)C)C)=O)(C)C CC(C)CCCCCC(=O)NCCCC(O)C(=O)NC1(c2nn[nH]n2)CC1 CN1CC2CCN(C(=O)CC3C4CCCC4N3C(C3(C(N)=O)CC3)=O)CC2C1 Cc1nc(C2(CN(C(=O)C(c3ccc(Cl)cc3)O)CC)CC2)cc(=NCC2CC2)[nH]1 c1(C(N2CC(CC(C(=O)N(CC)CC3CCCO3)F)C2)=O)cncnc1C C1(NC(c2cnc(C3CC3)s2)=O)COC2CN(C(C3(O)CCSCC3)=O)CC12 N1(C(c2ccc(C=C)cc2)=O)CC(C2CN(C(=O)C(N3CCC(C)CC3)=O)C2)C1 C#CCCC(=O)N1C(=O)CNC(=O)CCN(C2CC2)CC(CN(C)C)C1 C1(N(C(=O)CSc2cccnc2)C)CCCN(C(C2CCCNC2=O)=O)C1 c1(N(CCC)C)nc(=NC2CCCc3cn(C(C)C)nc32)nc[nH]1 N1(C(c2c(C)ncs2)=O)CCC2(CCC2CNC(C2COCCO2)=O)CC1 c12cccc(n1)C(=O)NCCC(=O)NC2.C1CC(=O)N1.NC(=O)OC c1(CC(N2C(CC(=O)OC(C)(C)C)CCC2)C(=O)O)ccc(F)cc1 C1(CC(=O)OC)CCC2CN(CC(c3oc(SC)nc3C)=O)CCC2C1 N1(C(C(C)NC=O)=O)CCC2CCCC12CNC(c1cc(C2CC2)ccn1)=O S(=O)(=O)(c1c[nH]c(C(=O)NCC2(OC)CCN(C(=O)CC(C)CF)C2)c1)NC c1(-c2nc(C(C)OCC)nn2CC2CC2)ccnc(CC)c1F C1(C(=O)NCC(C(C)C)(C)O)CN(C)CCN1C(=O)CCc1nc(O)n[nH]1 C(C(CC(=O)NC1CC(CNC(C2(C3CCCO3)CC2)=O)C1)C(F)F)N(C)C CCC(F)(F)C(C)(C)C(=O)NC1CC1NC(=O)C(C1CCOC1)OC C1(CNC(C(CC)(C)F)=O)CN(C(c2ccnc(Cl)c2N)=O)CCCO1 C1(CNC(c2c(OC)c(F)ccc2)=O)C(C2CC2)CCN1C(=O)CC1CCC1 N1(C(C2(CC)CC(F)(F)C2)=O)C2CCCC1CN(C(c1ncccn1)=O)C2 c1(C(=O)NCC2(C(C)NC(=O)C(C)(F)F)CC2)cc2ccccc2c(=O)o1 c1(C(=O)NCC(CNC(CCC(C)OCC)=O)O)cc2nc(C)[nH]c2cc1F C(=O)(CCC(C)CN(C)C)NCCNCCOCCCNC(CCCC(=O)OC)=O N1(C(Cn2c(C)cc(C(F)F)n2)=O)CC2(CCN2C(=O)COC2(C)CCCC2)C1 C(C)(CC(=O)NCCNC(c1cc2cc(Cl)cnc2o1)=O)(C(F)(F)F)N(C)C Cc1cc(C=CC(N2CC(n3cc(-c4ncoc4C4CC4)nn3)C2)=O)ccc1Br Cc1cc(F)cnc1C(=O)N(C)CC1CN(C(C2(CC(C)C)CC2)=O)C1 c1(SC)cc(N(C2CC(NC(C3CCCCN3C3CC3)=O)C2)C)nc(SC)n1 N1(C(C=CCOCCOC)=O)CCN(C2CCCC2NC(C2CC23CCC3)=O)CC1 N1(C(CSCCOC)=O)CCC(C(=O)NCc2n[nH]c3c2CCC3)C12CCC2 C1(NC(CC(CNC(=O)CCC(F)(F)F)OC)=O)CCOC2(CCC2)C1 C(=O)(N=c1cc(NC(=O)OC(C)(C)C)n(C)[nH]1)C1CC(C)S(=O)(=O)CC1 C1(C(=O)NCCN(C(Cc2cc(CC)no2)=O)CC)CCOC(C)(CC)C1 C1(C(N(C2CCCC2)CCOC)=O)CCN(C(C2COCC(C)O2)=O)CC1(C)C C1(C(=O)NCC2CCC(C)N(C(c3cncc(Cl)c3)=O)C2)C(O)C(=O)N(C)C1C c1(CC)nn(C)c(C(=O)NC2CC2CNC(c2cccc(C(C)(C)C)n2)=O)c1Cl C1(C)(c2ccc(C)cc2)CCCN(C(c2cnn(C)c2C2CC2)=O)C1 CCCC(CCC)C(=O)NCC1CC1CNC(C1(CCOC)CCCCCC1)=O c1(C(N2C(C)(C)CCC2)=O)nc2ccc(-c3ccc(F)c([N+](=O)[O-])c3)cc2s1 C1(COC)CN(C(c2cnn(C(C)C)c2)C(=O)NCC2CCCC2)C1(C)C c1(C(N2C3CC(NC(CC(C)(C)O)=O)CC2CC3)=O)ccc2c(c1)NS(=O)(=O)C2 Cc1nc2ccc(C(N3CC(NC(C4CC=CCO4)=O)CC(C)C3)=O)cc2s1 C1(NC(C2CCN(C(=O)CCc3ccco3)CCO2)=O)CC2CCC1(CO)C2 N1(C(Cn2c(C)nc(C)n2)=O)CCC(CNC(c2nocc2Cl)=O)C(C)C1 c1(C(=O)NC(C)C(CO)NC(c2cccc(Cl)c2)=O)ccc(CO)c(Cl)c1 C(C)(C)(C(=O)NC(C1CCCC1)CNC(c1coc(Br)n1)=O)NC(=O)NCCC C1(CC#C)(C(=O)NCC2CN(C(c3nncn3C3CC3)=O)C2)CCOC1 N1(C(c2cnc(Cl)[nH]2)=O)CC(NC(C2(c3cc[nH]n3)CCC2)=O)C(F)C1 C=CCCCC(=O)N(C)CC1(C)CCCC1NC(=O)C(C)C(F)F C#Cc1c[nH]nc1C(=O)NC1CCC(CCOCC2CCC2C(=O)OC)C1 C=C(C)CC(C(=O)NCC1CC(C)C1)NC(=O)CC#N c1(CN(C(C)C)CCN(C)C(c2cc(C3CCNCC3)no2)=O)ccccc1F C12(C(=O)NCCCN(C(C(C)OCC)=O)CCOC)CC(C)(C1)OC21CCC1 c1(NC(C2OCCN(C(C3(C)C=CCC3)=O)C2)=O)ccc2cnccc2c1 N1(C(C(P(C)(C)=O)O)=O)CC2CCN(C(=O)CN3CCc4ccccc43)CC2C1 N1(C(c2c(C)cnn2C)=O)CCN(C(C2CC(=O)N(CC(C)C)C2)=O)CC1C N1(C(C2(CC#C)CCCCO2)=O)CC2CCN(C(=O)Cc3c[nH]nc3O)CC2C1 C1(C(=O)NCCOCCNC(=O)C2=CCOCC2)C2CCC(C2)S1(=O)=O Cc1[nH]c(C#N)cc1C(=O)N(C(C)CN(C(=O)C1=NNC(C(F)(F)F)C1)C)C Cc1c(Br)csc1C(=O)NC12CC(NC(=O)CC3(C)CC3)(C1)C2 CC12CCC(C(=O)NC3CC(F)CN(C(=O)C=Cc4ccccc4F)C3)(CO1)C2 c1(C(=O)NCc2ccc(CS(C)(=O)=O)cc2)ccc2c(c1)-c1ccccc1C2 C(CC(C(=O)NC1(C)CN(C(=O)CCCF)C1)NC(=O)OC(C)(C)C)SC.C(N)(=O)N n1(CCc2cn(C3C(C)(C)COC3=O)nn2)cnc2ccccc2c1=O C(=O)(CC(C)(C)C1CCCCC1)N1C(CNC(C2N(C(C)=O)CCC2)=O)CC1 c1(C(=O)NCC2(CNC(CCCOCCOC)=O)CC2)ccc2cnccc2n1 C1(C(N(CC#CC)C)=O)CCCC(NC(c2cccc(C)c2F)=O)CC1 c1(C(=O)NC(CNC(=O)CCc2ccccn2)CO)ccc(O)c(F)c1F CC1CN(C(c2cc(Cl)no2)=O)CC1NC(c1cn(CC2CCOCC2)nn1)=O C(=O)(CC(CN(C)C)C(F)(F)F)NC1CC(NC(C2(NC(C)=O)CCOC2)=O)C1 c1(C(N2CCN(C(C=C(C)C)=O)C3(C2)CCC3)=O)cc(S(C)(=O)=O)ccc1Cl C(=O)(C1COc2ccccc21)N1C(C)CC2CN(C(C=C(C)C(F)F)=O)CC21 CC(C)(C)CC(O)C(=O)NCC(CO)NC(c1cnccc1Br)=O C(=O)(CC(C)(O)C(F)(F)F)Nc1cc(CC(=O)OCC)cc(O)c1 C1(CNC(C(OC)OC)=O)CC(O)C(O)CC1C(=O)NCC12CCC(F)(CC1)C2 C12N(CC13CCN(C(N1C(C(=O)OC)CCC1)=O)CC3)C(=O)NC2.C(C)(C)(C)O.OC CCC(C)C(O)CNC(=O)NCc1c(Cl)cnn1C C#CC1(NC(=O)CC(C(F)(F)F)NC(=O)Cc2ccccc2F)CC2CCCC12 c1(C(N2CC3C(NC(C4CC(CCO)C4)=O)(C3)C2)=O)ccc(Cl)c(F)c1F c1(C(N2C(C(=O)NC(CCC)CO)CC(O)C2)=O)cc(C)ccc1F CCC(Cc1ccccc1)C(=O)NCCC1(NC(=O)C=CS(C)=O)CC1 c1(NC(=O)NCC(F)C(=O)O)cccc(C(F)(F)F)c1Br CCCCC(O)C(C)C(=O)NC1CC(C(N2CC(N3CCCC3)C2)=O)C1 c1(C(C)C)ccc(C(=O)NC23COC(C2)C(NC(=O)C(F)C(C)(C)O)C3)cc1Cl c1(OCCOC)ccc(F)c(C(N2CCCC(c3n[nH]c(C4CC4)n3)C2)=O)c1O CC(=NO)C1CC(C(N2CC3CC2CN(C(=O)CN2CCC2)C3)=O)C1(C)C CC(C)CC(CNC(C1CCN(C(N)=O)CC1)=O)NC(=O)CCc1cccnc1Cl C(=O)(C(CC1CCC1)NC(c1cn(CC)cn1)=O)NC1(CCCC)CC1 CCS(=O)CC(=O)NC(C)C=CC(=O)NCC(C1CC1)SC N1(C(C2N(CC)CCC2)=O)CC(C)(C)CC1C(=O)NC1CC(OC)C1 C1(O)(C(=O)NC2C(CNC(c3c(C)ccc(C)n3)=O)CCC2)CN2CCC1CC2 CCCCCCC(C)CC(=O)NCC(F)CNC(c1c[nH]nc1[N+](=O)[O-])=O C(=O)(C1SCCc2ccccc21)NC1CCC(NC(c2cnc(CC)[nH]2)=O)CC1 N1(CC(=O)NCC(CC(=O)OC)(C)C)CCC2(CCC2)C(CO)C1 C12CCCN1C2=O.C(CC(=O)N(C1CC1)C)OCCOC.C1(C2CCC2)CCCO1 c1(CC)c(C(N2CCC(CO)C(NC(=O)C(C)(C)C#N)C2)=O)oc2ccccc12 CCC(F)(F)CC(=O)NC1CCC(CC(=O)N(C(C)CN(C)C)C)C1 C1(CC(=O)NC)CCCCN1C(CCC1CC(F)(F)C1)C(=O)NC CC(C)CC(C)C(=O)NC1(CF)CCN(C(c2ncccc2N(C)C)=O)C1 c1(N(C(C)=O)C)ccccc1C(N1CC(NC(C2CC(N(C)CC)C2)=O)C(O)C1)=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(NC(CCCOC(C)(C)C)=O)COC1 c1(C(=O)NC(C)(C)CCNC(=O)CNS(C)(=O)=O)ccc2nsnc2c1 C1(C(=O)OC(CCSC)C)CN(C(=O)NC(C)(C)C)CC12CC2 c1(C(=O)N(CCNC(C23CSCC2C3(F)F)=O)C2CC2)ccc([N+](=O)[O-])s1 Cc1c(Cl)ccnc1C(N1CCOCC1CCNC(=O)C(F)C1CCC1)=O c1(CCC)nnc(S)n1CC(=O)NCCC1CCN(C(c2cncc(O)c2)=O)C1 N1(C(C=CC2(C)COC2)=O)CCCC12CCN(C(=O)Cn1ncc(Br)n1)C2 C1(NC(c2ccc(C#C)o2)=O)CCCN(C(C2CCN(CCC)CC2)=O)CCC1 N1(C(Cc2n(C(C)C)cnn2)=O)CCN(C(c2cc(N)ccc2F)=O)C(C)C1 Cc1nc(C(=O)NC2CCC(NC(c3cncc(F)c3)=O)C2)c(C)o1 S(=O)(=O)(c1cc(OC)ccc1Cl)N1CCCC(C(=O)NCCC#C)C1 C=C(Cl)C(C)(C)C(=O)NCC(F)CNC(=O)C(c1ccc(F)cc1)(C)O Cc1nc2c(C(=O)NC(C)C(CO)NC(=O)C(C)(C)C3CCOC3)ccnc2[nH]1 Cn1ccc(C=CC(=O)NCC2(CNC(=O)CC3CCCCC3)CC(F)(F)C2)c1 n1(CC(=O)NC(CCNC(C(C2CCOC2)OC)=O)(C)C)nc(C)nc1C C(=O)(C(CO)C(C)(C)C)N1CCC(C(C(=O)Nc2c(OC)n(C)nc2)C)CC1 c1(C(=O)NCC23CC2CN(C(c2ccc(F)cc2F)=O)C3)ccc2nonc2c1 Cc1cc(C)n(C(C)C(=O)NCCN(C(=O)Cn2cncn2)C2CC2)n1 Cc1nc(CC(=O)NC2CCN(C(=O)C(n3cc(Br)cn3)C)C2)sc1C CN(CCC(=O)Nc1ccccc1F)N1CCCCC(O)C1 C(=O)(C1=CC2CCC=CCCC12)OC.c12cc(c(OC)c(F)c1)C(=O)N2 C1(CNC(C2(CC#C)CC2)=O)CCCCN1C(c1cnc(C(C)=O)s1)=O CC1(C)CN(C(=O)CCN(C(=O)Nn2cccn2)C(=O)CO)CCC1CO c1(C(C)C)cc(C(=O)NCC2CC(C)N(C(c3[nH]c(C)cc3C)=O)C2)c(CO)[nH]1 NS(=O)(=O)CCC(=O)NC1CN(C(c2cccc(N3CCNC3=O)c2)=O)C2CC12 N1(CCNC(c2c(C)noc2C(C)C)=O)CC(=O)N2CCCCC2C1 C1(NC(C=C(C)C)=O)C2CCN(C(=O)CCc3ccccn3)CCC12 c1(CC(C=C)CC)nc(-c2ccc(C)o2)nn1-c1cccc(C(F)(F)F)c1 N1(C(C(=Cc2cccs2)C)=O)CC(CNC(C2CCNC(=O)C2)=O)CC(C)C1 Cc1ccc(F)cc1NC(C1C2CCC(C2)C1NC(c1cc(F)n(C)n1)=O)=O c1(C(=O)NCC2C3CCCC2N(C(=O)CC)C3)cc2cc(Cl)ccn2n1 C1(NC(CC(CC)C)=O)CC2CCC1N2C(c1ccc(Br)cc1N)=O c1(C(N2C(CNC(=O)Cn3ccc(C)n3)CC(OC)C2)=O)ccn2nccc2n1 CC1(CNC(C2CC3(CSC3)C2)=O)CCCN(C(c2ncccc2C(F)F)=O)C1 C#CC1CC2(CC2)CN1C(C1CC(C)CN1C(C1CCC(C)(C)C1)=O)=O c1(CN2CCC(CNC(CCC(=O)NCC)=O)C2)ccc(Cl)cc1Cl N1(C(=O)CO)CCCC2(CCN(C(C3(Cc4ccccn4)CC3)=O)CC2)C1 N1(C(Cn2ncc(C)c2)=O)CCCN(C(c2ccc3c(c2)nnn3C)=O)C(C)C1 c1(C(=O)NC(CC)(CC)CCNC(c2cnn(C)n2)=O)cc2c(ccn2C)s1 CCCC(C)(CC)C(=O)NC1CC(O)CN(C(c2ccc(-c3ccco3)s2)=O)C1 C12(CNC(Cc3cc(C)nn3C)=O)CCC1CCN2C(C1(NC(N)=O)CC1)=O c1(C(=O)OC)[nH]ccc1CNC(c1cc(C)cs1)=O Cc1ccc(F)c(C(=O)NC(C2(O)CCCCC2)C(N2CC3CC(C)C3C2)=O)n1 N1(C(C2C(C)(C(C)C)C2)=O)CCC(C)(CC(=O)NC2C3CCC2CC3)C1 C(=O)(CCC1=NNC(=O)CC1)N1CC2C(CNC(C(C(C)C)NC(N)=O)=O)(C2)C1 c1(CC(=O)NCCN(C(=O)CCC2CNC(=O)N2)CC)cc(F)cc(F)c1 c1(C(=O)NC(CCNC(C2C(C)CC2C)=O)(C)C)cncc2sccc12 N1(C(c2c(CC)nco2)=O)C(C(N2CC3(CCCCC3)C2)=O)C2CC(O)C1C2 CC1CS(=O)(=O)CCCN1C(C1C2CN(C(c3cc(Cl)c[nH]3)=O)CC12)=O c1(C(N2CC(COC)C(C)C2)C(=O)NCC(=C)C)ccc(CC(C)C)cc1 N1(C(C(C)(C)CO)=O)CCC(n2cccn2)(CNC(=O)C=Cc2cncs2)CC1 CSC=CC(=O)NC(C1(O)CN(C(=O)C=CCN2CCCCC2)C1)C C(C)(CO)(C(=O)NCCC1(NC(c2ccoc2)=O)CC1)OC c1(N2CC3CC(NC(c4c(C)nc[nH]4)=O)CC3C2)ccc(C#N)cc1[N+](=O)[O-] Nc1c(C(N2CC3CC(NC(c4cc(CCO)on4)=O)C2C3)=O)ccc(F)c1F C(=O)(C(C)CC(C)(C)C)N1CCN(C(c2c(CCC)nsc2N)=O)CC1CCC C(=O)(C1CCCc2nc[nH]c21)N1CCCN(C(c2ccc[nH]2)=O)CC1CO CC1CC(C(N2CCN(CC(=O)N3CC(OCc4cccs4)C3)CC2)=O)CCO1 c1(COC)ncsc1C(=O)NC(C)CCCNC(c1[nH]cnc1C)=O C=Cc1cnn(C)c1C(N1CCCC(CC)(NC(C2CC2C2CCC2)=O)C1)=O N1(C(=O)OC)CCCC(n2cc(NC(=O)Nc3cnc(C)n3CC#N)cn2)C1 c1(OC)cc(C(=O)NC2CC(F)(CNC(=O)C(C)n3cccn3)C2)ccc1C N1(C(CNS(CC)(=O)=O)=O)CCC(C2(NC(C3CN(C)CC(C)O3)=O)CC2)C1 C#CC1CN(C(C23CCCCC2C3(F)F)=O)CCN1C(c1nc(CC)oc1C)=O CC1C(NC(C2CCSC(C)C2)=O)CCCN1C(c1cncc(C(F)F)c1)=O CCCC(C(=O)N1CC(CS(C)=O)C1)NC(c1cnn(C)c1Cl)=O C1(C(=O)OCC)CCc2sc(N3CCN(C4CCCCC4)CC3)nc2C1 C(CNC(=O)CCCN1C(=O)CNC1=O)(C(C)C(C)C)NC(c1cnc(C)o1)=O C(=O)(C1Cc2ccccc21)NC(C(=O)NC(C(CC)C)C(=O)NC)(C)CSC c1(C(N2CCC=C(C(=O)OCC)C2)=O)ccc2oc(O)nc2c1.C12CC1C(=O)N2 c1(C(=O)NCCN(CC(C)O)C(=O)C=CC2CC2)cn(C)nc1C1CCOC1 c1(C(N(CC(CC)NC(CCc2onc(CC)n2)=O)C)=O)ncnc(C)c1C N1(CC)CCCC1CNC(=O)CCN(C(=O)CNC(=O)CC1OCCCO1)C C1(N(C(=O)C2=CCCS2)C(=O)CC(=O)N2CCNCC2)CCCN(c2ncccn2)C1 CCC(C)CC(C)C(=O)NCC#CC(=O)NCc1nnn(C)n1 C(=O)(C1CCCc2ncnn21)N1CC(N(C(C2=C(C)OCCC2)=O)C)C2(C1)CC2 CCCCS(=O)(=O)NCC(=O)NC1(CCO)CN(C(=O)Cc2cnoc2)C1 c1(C(=O)OCC)cccc([N+](=O)[O-])c1NC(=O)NCC(N1CC2C(SC)(C2)C1)=O N1(C(C23CCC(OC)C2C3)=O)CCC2CN(C(c3c(O)nnc(C)c3C)=O)CC12 N1(C(C2(CC)CCCC2O)=O)CCn2ncc(CNC(=O)C=C(C)C3CC3)c2C1 c1(C(=O)NC2CC(OC)C2)cnc(SCCNC(c2cc(O)cs2)=O)nc1 C(C(C)(C)CO)(c1ccccc1)NC(C(Cc1ccco1)NC(C)=O)=O C1(NC(C2(OCC)CCC2)=O)CC2(C1)CC(C(=O)NC1(C)CCCC1C)C2 C(=O)(CCCC(C)CC)NCCCC#C.c1(C2C(=O)N2)cn(C)nn1 c1(C(=O)NC(CC2CN(C(C(C(CC)CC)C)=O)C2)C)[nH]c2ccccc2c1Cl C12(C(=O)NCC(C)NC(=O)CCC(=O)c3ccccc3)CCC(C(F)F)(CC1)C2 N1(C2N(C)C(=O)NC2)CCN2CCOCC2(CO)C1 C1(NC(=O)CCN2CCCC2)CCN(C(=O)CN2CCOCC2=O)CC1F C(CC)(CC(=O)NCCC(CC)CO)NC(COCCOCC)=O N1(C(CSC(C)(C)C)=O)CC(=O)CC(C(=O)NCC2CC2(Cl)Cl)C1 Cc1cccc2c(C(=O)NCCC(O)CNC(C3CC(O)CN3C)=O)n[nH]c12 C12(CNC(C3CC(OC)C3)=O)CCC(CN(C(C3COC4COCC34)=O)C1)C2 NS(=O)(=O)c1cc(Br)ccc1C(N1CCC(O)(CC(F)(F)F)CC1)=O C12COc3ccc(cc3C1)NC2=O.C1(O)(CF)CC(NC(CCSCC)=O)C1 N1(C(C2=C(C)CCC2)=O)CC(NC(c2csc(Br)c2)=O)CC12CCCCC2 c1(OC)cc(NC(C23CC2CN(Cc2ccc(Cl)o2)C3)=O)c(Br)cc1F O=C1CCc2cc(Cl)c(S(=O)(=O)NCC3CCCS(=O)C3)cc2N1 CC1(C(N2CCC(C(CO)NC(=O)CC3CC3)CC2)=O)CCNC(=O)C1 N1(C(C2(NC(C(C3CCC3)OCC)=O)CC2)=O)C2CCC1CC(O)C2 N1(C(c2occ(C)c2)=O)CCC2(C1)CN(C(c1nccs1)=O)CCO2 C(C)(N=c1nc2c(cnn2C)c(NC2CCN3CCCC3C2)[nH]1)c1cncc(C)c1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2(CC(NC(c3ccc(C(F)F)s3)=O)CO2)C1 c1(C(=O)NCC2(CN(C)C(C3CN4CCC3CC4)=O)CC2)cnc2n1CCOC2 c1(C(N(CCCNC(C2CCC2F)=O)CC)=O)nccnc1Nc1ccccc1 Cc1noc(C)c1CC(=O)NC(C)(C)CNC(=O)C(C)NC(N)=O C(=O)(C(C)(C)O)N(C(C(=O)NCCc1ccon1)C1CC1)C N(C1CCc2ccccc21)(CCCOCC)Cc1ccc2nc(O)oc2c1 c1(SC)cc(C(N2CCC(CO)C(NC(C3(C#N)CCCC3)=O)C2)=O)ccc1F C(=O)(C(C)(C)C(O)C(C)C)N1CCC2CN(C(CCCCCOCC)=O)C2C1 C1(F)(CN(C(C2N(C(CC)=O)CCC2)=O)C2CC2)CCN(C(=O)C#CC(C)C)C1 c1(SC)ncc(C(N2CC(O)CC2CNC(=O)COC(F)(F)C(F)(F)F)=O)cn1 c1(C(N2C(C)CC(CNC(CC(=O)OC)=O)C2)=O)cnc(O)c(C)c1 N1(C(COC2CC(NC(C3C(OC)CCC3)=O)C2)=O)CC2(C)CCC2(C)C1 C1(C(N2CCN(C(Cn3c(C(F)F)cc(C)n3)=O)CC2)=O)CN(C)CCN1C C1(CNC(CN(C2CCC2)C)=O)CCC(O)C1.C12CCC1NC2=O C(C(C(=O)NCCOCC(C)(C)O)n1cc(C2CC2)nn1)OCC.C(CC(=O)O)CC n1(CC(N2CCC(C)C2CNC(=O)COC2CC2)=O)ccc(O)nc1=O c1(CC)ccc(C(C)F)cc1.C12(C)CC(C1)NC(=O)C1CC(C1)OCC(=O)N2 c1(C(N2CCCCC(CNC(C(C)SCC)=O)C2)=O)nc2ccccc2nc1C C1(NC(C2N(C)CCCC2)=O)CN(C(c2ccnc(F)c2N)=O)C(C)(C)C1 N1(CCNC(=O)C(=O)NCC2C3COCC23)CCc2ccccc2C1 Cc1cc(Cl)c(F)cc1NC(=O)CN1CCOCC1.C12CC1NC2=O C1(O)(CNC(=O)Cn2ccnn2)CCOCC1.n1(CC(O)C2CC2)cccc1 c1(N(C2CC(OC)C2)CC2CC2)cc(C)c(S(=O)(=O)NC2CCOC2C)cn1 C1(C(N2CC(C(=O)OC)(OC)C2)=O)CCN(S(=O)(=O)C(F)(F)F)CC1 S(C1=NS(=O)(=O)c2ccccc21)CCNC(C(C)CC(C)(C)C)=O Cc1ccn2cc(C(=O)NC3CC(NC(C4(C)CC4Br)=O)C3)nc2c1 C1(C(=O)NCC2CCN(C(=O)Cc3cccc(O)c3F)C2)CCN2CCOCC12 S(=O)(=O)(c1ccc(C)c(C)c1)N1CCN(C(C(C)=O)=O)C2C1C2 CCC(C(=O)NCC1(F)CN(C(=O)C(C2CCCCC2)OC)C1)OC O=C1Cc2cc(C(=O)NC3CC4CN(C(c5cnccn5)=O)CC34)ccc2N1 N1(C(CCS(=O)(=O)NC)=O)CCCCC(CNC(=O)C(F)C(F)(F)F)CC1 c1(NC23C(CN(C(C(C)OCC=C)=O)C2)CC3)cccc(F)c1C#N c1(OC)ccc(C)c(C(=O)NCC(CO)NC(C2COCC2(C)C)=O)n1 Cc1cnccc1CN(C(=O)C(Cn1ccnn1)NC(=O)CN1CCNC1=O)C C1(C(N2C(C3(O)CN(C(C=CCOC)=O)C3)CCC2)=O)CCC(C)(CC)CC1 N1(C(C2N(C(CNC(=O)OCC)=O)C3CCC2C3)=O)CCOCC2(CCC2)C1 c1(C(=O)NC2CCN(C(C(C(C)C)n3cc(C)nc3)=O)C2)ccnc2cc[nH]c12 C(=O)(CC(C(C)CC)NC(=O)CCCC(C)=O)NCC1CCN(CC)C1 N1(C(CSc2nc(C)[nH]n2)=O)CCC(C)(C)C1CNC(=O)CN1C(=O)CCC1=O n1(C(C)C)ncc(C(=O)N(C2CCCC2)CCNC(c2coc(Cl)c2)=O)n1 n1(CC(=O)NCC(C)(C2CC2)NC(C(C)C2CCC2)=O)cc(Br)c(=N)[nH]1 C(=O)(C#CC1CCCCC1)N1C(C)CCN(C(=O)Cn2ncccc2=O)CC1 c1(-n2c(C(=O)NCC3C(CNC(C4(S(C)=O)CCC4)=O)C3)cnn2)ccc(Cl)cc1 C1(NC(C(c2ccncc2)C)=O)CCC(C)N(C(C2C3C4CCC(C4)C23)=O)C1 N1(C(C=Cc2cc(OCC)ns2)=O)CC(C)CN(C(=O)CCCC(N)=O)CC1C c1(CNC(=O)NCC(c2cccc(Br)c2)(C)O)nc2c([nH]1)CCCC2 N1(C(C(C)CC(F)F)=O)CC2CC(C1)CN(C(=O)C=Cc1ccc(C(F)F)o1)C2 c1(C(C)OCC)noc(CNC(=O)C(C)C2CN(C(=O)CCCSC)C2)n1 CC1(C)CC(CC(N2CC(c3ccccc3)(NC(c3csnn3)=O)C2)=O)CO1 C1(C(=O)NCC2(OCC)CC2)CCC=CC1CNC(=O)CC n1(CC)ncc2cc(C(N3CC4CCC3CN4C(c3csc(Cl)c3)=O)=O)cnc12 N1(C(c2c(OC)nccc2)=O)C2CCC1C(C)C(NC(=O)CCc1cn[nH]c1)C2 N1(C(C(=O)OCCN2CCOCC2)=O)CCc2sccc2C1.c12ccc(cc1)s2 N1(C(C2(C)CCCO2)=O)CC2CCC(C1)C(NC(=O)CC1CCCC(=O)C1)C2 C(CC1CC1)(C(=O)NNC(=O)C1(N2CCCC2)COC1)NC(=O)OC(C)(C)C C(=O)(CCCCCC(C)O)N1CCC(NC(c2cc(OC)c(C)cc2)=O)(CF)C1 CC1CN(C(c2cccnc2SC(F)F)=O)CCC1CNC(c1csnc1Cl)=O Cc1cc(C)c(C(=O)NC2CC(C(C)NC(=O)C(O)c3ccsc3)C2)c(N)c1 c1(OCC#C)ncccc1C(=O)NCC(CO)NC(=O)C(C)CC=C C(CCN=c1[nH]c(=NC2CCCN(C(=O)N(C)C)C2)[nH]c2c1COCC2)SC N1(C(CN(CCOC)C)=O)CC2(CCCC(CNC(c3n[nH]c(C)c3C)=O)O2)C1 C1(O)CCN(C(C2(C3CC3)CCC2)=O)CC1.C(CC(=O)NC)OCCC N12CCOC(C1)C2=O.C1(CN(C)C)CC(=O)N(CC)C1.C(CCO)N(CC)CC N1(C(=O)Cc2ccc(Br)nc2)CC2CCN(Cc3cnc[nH]3)CC2C1 c1(C(N(C)CC2CN(C(=O)CC3CC3)C2)=O)cccc(I)c1 N1(CC(=O)N(CCC(C)NC(=O)C=C2CCC2)C)CCCC(C(F)(F)F)C1=O c1(C(N(C(C=C)C)Cc2ccccc2)=O)cccc(-c2cncnc2)c1 C1(Sc2ccccc2)CCCN(C(=O)CCCCn2cc(-c3occc3)nn2)C1 c1(CC(=O)NCC(C)(C2CC2)NC(=O)C=C2CCCC2)c(F)cncc1Cl C1(NC(c2c(C)scn2)=O)CCCCC1NC(=O)CCCN(C)C(C)C c1(C(=O)NCC(CCNC(c2c(C)cncc2)=O)O)cccc(N=S(C)(C)=O)c1 N1(CCNC(C2(C(C)C)CCCO2)=O)CCN(C(C2CCC2(F)F)=O)CC1 N1(CCC)CC2CCC(C1)N2Cc1ccc(O)cc1 C1(C(CNC(C=C(C)C(C)(C)C)=O)C)CCN(C(C2(CF)COC2)=O)CC1 CC(C)CC(O)C(=O)N1CCC(CC(=O)NC2CNC(=O)C2)CC12CC2 C(=O)(C1=NOC(C)C1)NC(c1nc(C(=O)NCCn2ncccc2=O)co1)C C1(NC(=O)C=CBr)CCOC12CCN(C(c1c[nH]nc1C1CC1)=O)CC2 Cc1cc(CN(C(=O)COC2CCN(C(=O)Cc3csc(C)n3)C2)C)no1 c1(N(C(C)=O)C2CC2)nn(C)cc1[N+](=O)[O-].C1(N)CCC(C)N(C(C2CC3CCC23)=O)C1 N1(C(C23C(CN(C(C(C)Cc4ccccc4)=O)C2)C3)=O)CCc2sccc2C1 c1(C(N2CCC(CCNC(c3cncc(C(N)=O)c3)=O)C2)=O)ccc(N)cc1F CCCCC(C)C(=O)NC1CCN(C(c2cc(O)cc(F)c2)=O)C1C1CC1 CCC(C)CCC(O)CC(=O)NCC(C)NC(c1ccc(C(C)(C)C)c(Cl)c1)=O C=CCCCC(C(=O)N1CCCC(CCF)C1)NC(c1n[nH]cc1C#C)=O C1(NC(Cc2ccc(C)nc2Cl)=O)C2CCCCN(C(=O)C(F)C(C)C)C12 c1(OC)cc(C)c2cc(C(=O)NC3(CF)CCN(C(C4CCOC4)=O)C3)[nH]c2c1 CCCCCCCCC(=O)N1CCC(O)C(NC(=O)C(CC)CC)C1 C1(NC(c2scc(C)c2C)=O)COC2C(NC(c3ccnc(C)c3C)=O)COC12 c1(CCCC(=O)NC2(CNC(=O)Oc3ccc(F)cc3)CCC2)ccccc1Cl C1(CNC(c2c(CC)scc2)=O)COCCN(C(=O)CNc2ccccc2C)C1 CC1CC(CNC(=O)CC(C)(C)c2ccccc2)CCN1C(c1nccn1C)=O C(=O)(CC=C(Cl)Cl)NC(C(=O)NCC(C)F)c1cccs1 N1(C(C2=C(C)CC2)=O)CC2(CC(NC(c3cccn3-c3ccccc3)=O)CO2)C1 N1(C(C(C)OC2CCCC(=O)C2)=O)CC2CCN(OC)CC12 c1(CC)ccc2cc(C(=O)NC3CCCC(NC(=O)COCCF)C3)ccc2c1 CC1(C)CCCOC1C(=O)NCCC1CCC(NC(c2cnc(O)c(F)c2)=O)C1 N1(C(C2C(=C)CC2)=O)CCCCC1CNC(c1ccn(-c2ccc(O)cc2)n1)=O Cc1c[nH]c2cc(C(N3CC(F)(CNC(C4CC4F)=O)C3)=O)ccc12 CCCCC(C)N(C(=O)CCC1CCN(C(=O)CC2(OCC)CC2)C1)C.OCC C(=O)(CC(C)C(F)(F)F)NC1CC(C(=O)Nc2nc(C)sc2)CC1O c1(C(=O)NCC2CCCN(C(CC3CCC(C)C3)=O)C2)cc(O)cc(C#N)c1 N1(C(C2CC(C)(CC)OCC2)=O)CCC2CCN(C(c3coc(CC)n3)=O)C2C1 c1(C(=O)NC2CC(NC(=O)C(c3ccccc3)=O)C2)ccc(F)c2cccnc12 N1(C(C(C(C)NC(=O)COCCCF)C)=O)CC2(CNC(=O)C2)C1 N1(c2[nH]c(=NCC34CCC(CC3)C4(C)C)cc(C)n2)CC(O)C2(CCOCC2)C1 C1(C)(CNC(CC2(COC)CC2)=O)COCCN(C(C2CCC(F)(F)C2)=O)C1 c1(C(=O)NCC2(F)CCCN(C(CCC=C)=O)C2)nccn2nc(C)cc12 C(=O)(C(C)CC(F)F)NC(C(=O)NCc1cnc(COC)[nH]1)C1(C)CC1 c1(C(=O)NC(CC(C)C)CNC(=O)C=Cc2ncc[nH]2)cc2c[nH]nc2s1 n1(CCOC)nnnc1C(CCC1CCCC1)NC(COC)C1CCC1 CC(=O)CCCC(=O)N1CCC(NC(c2cc(OC(F)F)cc(F)c2)=O)C(F)C1 c1(C(N2CC3C(CNC(=O)CC4CCOC4)C3C2)=O)nnc(O)c2c1CCCC2 c1(OCCC(=O)NC2(C(=O)NC3CC(CSC)C3)CCC2)ccccc1Cl c1(CC)ccc(C(=O)NCC2(NC(=O)CCc3ccc(Br)cn3)CC2)cc1 c1(C(=O)NCC(CC)NC(c2ncnn2CC)=O)cccc(C(N)=O)c1C c1(CC(=O)NCC2N(c3c(C(=O)OC)cncc3)CCC2)cn2cc(C)sc2n1 c1(C(=O)NC2CC(C)N(C(=O)Cc3ccccc3)C2)cnc2ccnn2c1O c1(C(C(=O)NCC(C)CNC(C2CC2(C)C(F)(F)F)=O)F)ccccc1 N1(C(c2c(OC)csc2)=O)CCC(C)(C)C1C(=O)NCC1(C)CC(O)C1 c1(C(N2CCCC(CSCC)C2)C(=O)N(C(C)C)C2CC2)nc(Br)ccc1C C1(C(=O)NC(C(CC)C)CO)CC12CCN(C(=O)C(c1cccc(O)c1)C)CC2 c1(C(C(N2CC3C(CNC(C(C)N(C)C)=O)C3C2)=O)C)ccc(F)c(F)c1 CC1CN(C(=O)CO)CC1(C)C(=O)N(c1cnn(C)c1C(N)=O)CCC(F)(F)F Nc1cc(C(N2CC3CC2(C(=O)NC2(C4CCCO4)CCC2)C3)=O)cc(F)c1 N1(C(c2c(OC)n[nH]c2)=O)CC(NC(=O)C(F)(F)C2CCCC2)C(O)C1 c1(OC)ccccc1S(=O)(=O)Sc1ccc(-c2ccnc(SC)n2)s1 c1(C(=O)NCC2(OC)CN(C(=O)CSC(C)C)C2)csc2c1CCCC2 N1(C(CCOCCC)=O)CCCC(CNC(=O)COCC(=O)OC(C)(C)C)CC1 C(=O)(CCCCCF)NC12CC(C(=O)NCC3N(C)C(=O)CC3)(C1)C2 CC1CN(C(=O)CCC2(C#N)CCC2)CC(C)CN1C(c1cnc(N(C)C)o1)=O C1(C(=O)NC(C(C)C)(C)CNC(c2cnn(C)n2)=O)Cc2ccccc2C1(C)C C1(CC(N2CCC(NC(C3CCC(F)(F)CC3)=O)C2)=O)CC2(CCCC2)CO1 N1(C(CCCCCC=C)=O)CC2CC(C)N(C(=O)C(F)n3ccnc3)C2C1 C(=O)(C(CO)C(F)(F)F)N1C(Cn2cc(CCC(C)=O)nn2)C=CC1 Cc1oc(Cl)nc1C(=O)N(C(CNC(c1nc(=O)n(C)[nH]1)=O)C1CC1)C N1(C(C(=O)NC2CCOC2)C2CC2)CCC2(CC1)CC2(C)CO.CS c1(C(=O)NC2C=CC(C(=O)NCC(C)(C)C)C2)cc2cccnn2n1 C(=O)(CCC(C)NC(=O)CN(C)CCOC)N(CCC#C)C N(C1CCc2ccc3c(c21)CCO3)CCn1c(C(CC(C=C)(C)C)OCC)nnn1 C1(C(=O)Nc2cccc(Cl)c2)CC12CCN(C(c1c[nH]nc1C(F)F)=O)C2 c1(C(c2nnnn2-c2cccc(OC)c2)NCCCCOC)sc(C)nc1C C1(C(=O)NCCSCC2CC2)CNCC12CCCCCC2 C(CSC)(C(=O)C(=O)NC(C)CN(C(=O)CC1CCC(C)C1)C)OC.C(C)(C)(C)O CC1(F)CN(C(c2ccc3c(c2)CCCN3)=O)CCN(C(C2CSC2)=O)C1 n1(CC(=O)N(C2CC(NC(c3cc(O)ncn3)=O)C2)C)cc2ccccc2n1 C1(C(N2CCC(C)(CC(=O)Nc3ncccc3OC)C2)=O)(OCC)CCOCC1 c1(C(=O)NC2C(NC(CCc3n[nH]c(=N)s3)=O)CCC2)ccc(CC(N)=O)cc1 C1(CC(=O)NC2CC(N(C(=O)CC3C=CCCC3)C)C2)CCCNC(=O)C1 c1(C(=O)NC(C(C)NC(c2cc(N)cc(F)c2)=O)CO)cncc2ccccc12 C(=O)(C(COC)CC(C)C)N(CCCCN(C(CCC#CC)=O)C)C C1(COC)COC2(CCN(C(c3ccnnc3)=O)C2)C1.C123CC(C1)(C2)C(=O)C3=O N1(C(c2c(OCC=C)cccc2)=O)CCC(C=C)(C(N2CCCC2CF)=O)C1 CC1CCc2cc(C(=O)NC3CC(NC(=O)C(F)n4cccn4)C3)ccc2N1 C(CC(O)CO)N(C(C1(CCNC(C(C)n2cccn2)=O)CC1)=O)C C1(N(C(c2cc(C)n(C)c2)=O)C)CCC2CN(C(c3ccc(O)nc3)=O)CC12 Cc1cc(C(=O)N(C2CN(C(C3CC3C3CCCO3)=O)C2)C)sc1C N(C(=NCC=Cc1ccccc1)N1CCC(F)C1)CC1(C)CCC(=O)N1 CC(C)CCCC(C)C(=O)NC(C(=O)NCC1(C)CCCCC1)C(C)(C)O N1(C(CCc2cc(C)n(C)n2)=O)CCC(NC(C2CC(O)C2)=O)C1(C)C C1(C(=O)NCCOCCCNC(C2C(C(=O)OC)OCC2)=O)CC1C1CCCC1 C1(C(=O)Nc2cccc(NC(Cc3n(C)ncc3Cl)=O)c2)CCC(C)(C)OC1 c1(NCc2c(OCC)nccc2)ccc(S(=O)(=O)NC2CC2)cc1 N1(C(CCC(=O)NCC)=O)CCC(C(N2CCC(C)(CO)C2)=O)C(O)C1 c1(OCCC(=O)NCC(C2CC2)NC(CSCCC)=O)ccc([N+](=O)[O-])cc1 C1(CCC(=O)N(CCOCC=C)C)CCCCN(C(C2(C)CCC3CC3C2)=O)C1 N1(CCNC(Cc2ccn(CC)n2)=O)CCCN(C(C2CC23CCCC3)=O)CC1 N1(c2nccc(N)c2Cl)CCc2ccc(Cl)nc2C1 C(CC(=O)NCCCSCCO)N(C(=O)CC1(C)CCC1)CC C(=O)(C1CCCc2nn(C)cc21)N(C(C)C(F)(F)F)C C1(O)(C(CNC(c2n(CC)nnc2)=O)C)CCN(C(=O)CCC2CC(F)(F)C2)C1 N1(C(c2c(C)ccs2)=O)CCC(NC(=O)CCc2nccn2C)C12CCCC2 CCC(CC(=O)N1CC=CC(C(N2CCC(CC3CC3)CC2)=O)C1)C(C)(C)C N1(C(C(CC(C)C)O)=O)CC2CC(NC(c3ccc4cccnn34)=O)CC1C2 CCC(COCc1csc(Cl)n1)(c1nnnn1C(C)C)Sc1ccccc1 C(=O)(CCCCCSC)NCCC1(C(=O)NC(CCC)C(=O)OCC)CCCC1 c1(C(=O)NC(CCN(C(C2=C(C)CCC2)=O)C)C)ccc(Cl)cc1[N+](=O)[O-] O=C(CC1OCCc2ccsc21)NC1=NCC2(CCOC2)N1 C1(CNC(C2CC(=C)C2)=O)CN(C(c2cc(F)c[nH]2)=O)CC1(F)CO N1(C(C2CC(C)(C(=O)OC)C2)=O)CCN(C(c2cccc(=O)o2)=O)C(C)C1C C1(N(C)C(c2occc2-c2cnn(C)c2)=O)CCN(C(c2ccnc(S)c2)=O)CC1 C(=O)(C1CCCn2cncc21)NC1(C2CN(C(C3CC(=O)NC3)=O)C2)CC1 c1(C(=O)NC(C(C(C)C)NC(=O)CCCCCF)C)cccc2ncnn12 C12(CNC(c3cnc(-c4ccccc4)o3)=O)CCC1CCN2C(c1ccco1)=O N1(C(Cc2c(CC)con2)=O)CCC(CC)(NC(=O)CC2CCC(F)(F)C2)CC1 C1(NC(C2(O)COC2)=O)C2CCC1N(CC1C(C)(C)C(Sc3ccccc3)C1)C2 c1(NC(c2cc(OC)c(OC)cc2)=O)ccc(S(=N)(=O)N(C)C)cc1 c1(C(=O)NC2(CNC(CS(N)(=O)=O)=O)CCC2)ccc2c(c1)COCO2 O=C(O)CCC(Cc1ccccc1)NC(=O)Cc1ccc(C(F)(F)F)cc1 N1(CC(=O)NC(CCNC(C(C)NC(CC)(C)C)=O)C(C)C)CCC(=O)NC1=O C#Cc1ccc(C)c(NC(C2CCCN(C(=O)CC3CCC(=O)N3)CC2)=O)c1 N1(C(CC=CCc2nc(C)sc2)=O)CCCC(n2cc(CC(=O)N(C)C)nn2)C1 CC(C)CN=C(NCc1ccccn1)N1CC2CCCCC2C1 C1(CCNC(C2(C)CCCC2)=O)CCCN(C(C2(CF)CC(F)(F)C2)=O)C1 c1(C(=O)NCC(C2CC2)NC(C(c2c(C)n[nH]c2C)C)=O)cnn2cnnc2c1 Cc1nc(O)nc(C)c1CC(=O)NC1CCCC1NC(C1CC12CCCCC2)=O CC1CCCN(C(C2(n3cnc(=N)[nH]3)CC2)=O)C1.C12CC(C1)C(=O)NC2 c1(NCCCNCC(F)(F)F)nc(N2CCC3(CCSC3)C2)c2ccsc2n1 N1(C(C(N2CC(C)(NC(C(N3CCOC3=O)C)=O)C2)=O)C)CCc2ccccc21 C1(C)C2Cc3ccccc3C12.c1(-c2cn(CCNC=O)nn2)cccc(OCF)c1 C1(CN(C)C(C2CCOC2(C)C)=O)CN(C(C2(CCF)CCOCC2)=O)CCO1 c1(C(C(=O)NC(CCCNC(COCCOCC#C)=O)C)C)cccc(Cl)c1 C1(CNC(Cc2c(C)cccc2)=O)CCC2(CO1)CC(NC(=O)CC1CC1)C2 C1(CCNC(COC)=O)COCCN1C(=O)CC1CC(OC(C)(C)C)C(O)C1 c1(C(C)(C)C#N)cc(C(=O)O)cc(CN2CCOCC2)c1 Cn1ncc(I)c1-c1cccc(CNC(=S)NCCCF)c1 c1(NC(C2(OC)CC(C(C)C)C2)c2nnnn2C(C)C)nc2ccc(OC)cc2[nH]1 N1(Cc2ccc(OC)nc2)CCC2(CC1)CC2C(=O)NC(c1cccc(Cl)c1)C N1(C(c2cc(C)cc(N)c2)=O)CC2CN(C(=O)CCC3CCN(C)CC3)CC2C1 C=C(F)C1(CC(=O)NCC(C)NC(c2c(OC)noc2C2CC2)=O)CCOCC1 CC(C)(C)C(CO)C(=O)N1CCCC(C(=O)NCC(c2ccco2)O)CC1 N1(C(C2C(C)C2)=O)CCC(C)(NC(c2cc(C(F)(F)F)ncn2)=O)C1 c1(CC(=O)NCC2CN(C(Cn3cnc(=N)[nH]3)=O)CC2O)c[nH]c2cccnc12 N1(C(CC2ON=C(CC)C2)=O)CCC(CNC(c2cnc(O)n2C)=O)C1(C)C c1(CNC(CC(C)C)=O)ncccc1C(=O)NCCCn1ccnn1 N1(C(C)=O)CCOCC(F)(CNC(=O)CCCCC(N)=O)C1 CC1OCCC1CC(=O)NCCc1ocnc1CNC(=O)CCN(S(C)(=O)=O)C Cc1nc(C2CC2)ncc1C(=O)NC(C)(C)CNC(C1CCCCS1)=O CCC(C(=O)N(CCC(=O)N(C)C)C)NC(=O)C(C)CO N1(C(C(c2ccccc2)=O)=O)CC2CN(C(c3cnc(F)c(Cl)c3)=O)CC2C1 C1(CC)C(=O)NCCN1C(=O)NCC1(CO)CC(C)(C)C1.c1(N)ccccc1 S(=O)(=O)(c1cc(Cl)ccc1Cl)N1C2CC(NC(=O)CCN3CCOC3=O)C(C2)C1 N1(C(CCCN(C)C(c2ccccc2)=O)=O)CCCC(N(C)C(C2COC2)=O)C1 C1(C(=O)OC(=O)NCc2c(CCSC)ocn2)CCN(CC)CCO1 N1(C(C(CC)n2cncn2)=O)CCC(C)(CCNC(c2cncc(N)n2)=O)C1 c1(C(=O)NCCCCNC(C23CCCCC2C3)=O)c(O)cc(F)cc1F N1(C(c2ccc(C)o2)=O)CC2CCCC2(NC(=O)COCc2ccccn2)C1 C(=O)(CCS(N)(=O)=O)NCC1(F)CN(C(COCCC)=O)C1 c1(C(N2CC(CC(=O)NCCC3CCO3)C2)=O)ncc(F)cc1F N1(C(C2(C)N(C)CC(OC)C2)=O)CCOC2(CCN(C(c3cnsn3)=O)CC2)C1 CSC1=C(C(=O)N2CCC(CNC(=O)C(F)F)C(C)C2)CCCC1 N1(C(CC2CC(CC)C2)=O)C2CCC1CN(C(=O)COc1ccc(F)cc1O)C2 c1(NC(CCC=C)c2nnnn2CC)cc([N+](=O)[O-])c(C)cc1C c1(C(N(CCCOCCNC(C(C)SC)=O)C)=O)cnc(C(C)C)nc1 c1(C(N(CC(CN(C(=O)C(F)n2ccnc2)C)O)C)=O)cc2cc(Cl)ccc2[nH]1 C1(C(=O)NCC2OCCN(C(c3c(C#N)cn[nH]3)=O)C2)CCc2ncnn2C1 N1(C(C(=O)NCCNC(C(CC)C)=O)=O)CC=C(C(=O)OC(C)(C)C)C1 C(=O)(CCCS(=O)(=O)N1CCCC1)NCCNC(c1ccccc1CSC1CC1)=O CN1CCC2C1CCCN2C(c1ccc(Cn2cc(C3CC3)nn2)o1)=O C(=O)(CCCCCC(=O)NCC1CCN(C(C2CCC2C)=O)CC1)OCC C1(NC(C=NOC)=O)CC2CCC1C(NC(C1(OC)CCC(C)(C)C1)=O)C2 N1(CC)CC(CNC(C2CCCC(CNC(C3CCCCC3C)=O)C2)=O)OC1=O c1(NC(c2c(C)nc(NC(CC=CCC)=O)s2)=O)cnc(O)c(Br)c1C C=CCC(CC(C)C)C(=O)NC1CCN(c2cc3nncn3cn2)C1 C1(C(N(C2CCN(C(c3cc(C)n(C(F)F)n3)=O)C2)CCC)=O)CC(F)CN1C C(=O)(C(C)(C1CC1)N)C(=O)CN1CCSCC1.C(C(C)N)(C1CCC1)OC CS(=O)c1ccccc1C(=O)NC1C2CC1N(C(C1CC1(F)F)=O)C2 n1(CC(=O)NCC2CCCC2C(=O)NC2CCCCC2O)c(O)nnc1O C1(C(=O)NC2CN(C(c3c(C)cc(F)s3)=O)CC2C)OCCCC1(C)C c1(CC)onc(C(=O)NCC2CCCN2C(c2ncc(Cl)s2)=O)c1C c1(CC)[nH]c(=NCC(F)c2ccc(Br)cc2)nc2c1cnn2C(C)(C)C C1(C)(C(N(CCCC)CCCC)=O)CC(O)CN1C(=O)C(C)Cn1cccn1 N1(C(c2c(C)occ2)=O)CC(NC(=O)C(C)(O)C(C)C)CC(F)C1 C1(c2n(-c3c(CC)cccc3)nnn2)(NCCOC2CCOC2)CCN(C)CC1 CCC(C)C(O)C(=O)N1CCC(CNC(c2ccc(Cl)cc2OC)=O)C1(C)C N1(C(C2(CC)CCOCC2)=O)CCC(CNC(c2cc(N)c(Cl)cn2)=O)CC1C c1(C(N2CCC(NC(C3C(C(N)=O)C3)=O)C(F)C2)=O)ccc2oc(S)nc2c1 N1(C(CN(C2CC2)CC)=O)CCC(NC(C2(C#N)CC23CCC3)=O)C(C)(C)C1 C12(C(=O)NC(c3ccccn3)CC)CC(CO1)N(C(=O)OC(C)(C)C)C2 Cn1nc(C(N2CC(OCC(=O)NC3CCC(CO)C3)C2)=O)cc1C1CC1 C1(C(N2C(CNC(=O)Cc3cc(Br)cs3)CCC2)=O)CC2(CCC2O)C1 Cc1csc(C(C)C(=O)NC2CC(NC(=O)C(C)N(S(C)(=O)=O)C)C2)n1 c1(C(=O)NCCC2OCCN(C(CCC(=C)Cl)=O)C2)cc(F)c(F)cc1Br C(C(N=[N+]=[N-])C(=O)NC(C(=O)NCc1ccccc1C#N)C(C)C)OCC c1(NC2C(C)CN(C(=O)CN(c3ccccc3)C)C2)ccnc2ncnn12 C1(C(C)C)CN(C(N2CC(OCC(C)(C)O)C2)=O)c2ccccc2O1 N1(C(C2C(C)(C(C)C)C2)=O)CC2CCC(C1)N2C(c1ccnn1C)=O c1(CNC(C2CC(C)OC2)=O)ccc2c(c1)CN(C(c1ccsc1)=O)C2 c1(CN=C(N(C)CC(C)C)N)ccc2c(c1)C(C)CC(=O)N2C.c1(CC)cccs1 N1(C(CCC2(N(C)C(c3ccccc3C#N)=O)CCC2)=O)Cc2ncsc2C1 C1(O)(C(C(=O)N(C(C)C(=O)NCCn2cnnc2C)CC)C)CCCCC1 C(=O)(C(O)C1=CCCCC1)NCc1ccc(CN(C(CCC(C)C)=O)C)cc1 N1(C(c2c(CCC)[nH]cc2)=O)CC(C)(C)CC1CNC(C1CCCC(F)(F)C1)=O O(NC(=O)C(CNC(=O)C(C)c1ccsc1)OC)CC=C.N(C)C C1(C(N(CCNC(c2cc(Cl)ncc2O)=O)CC2CC2)=O)CCC2(CCC2)C1 C12CC(N(C(=O)CCc3nncn3C)C1)C2.n1(CCOC)cc(C(C)OC)nn1 C1(C(N(C)C)=O)CCN(c2cc(NCC3CCN(C(C)(C)C)C3)ncn2)CC1 N1(C(C23CCN(C(CNC(=O)OCC)=O)C2CCC3)=O)CCC(O)CC(C)(C)C1 Cc1c(C(=O)NC(C)CNC(=O)C(N2CCCCC2=O)C)c(Cl)nn1C C(=O)(CCCCCCS(N)(=O)=O)N(CC(C)NC(C(CCC)C(C)C)=O)C c1(OC)nc(C(N2CCCC(CNC(=O)CC(C)(O)COC)C2)=O)cc(O)n1 N1(C(c2[nH]cc(CN(C)C)c2)=O)CCCN(C(=O)CC2CCCC2O)CCC1 N1(C(C2N(C(Cc3scc(C)c3)=O)CC(O)CC2)=O)CC2CCC(O)C2C1 Cc1cccc(C(=O)NCCNC(=O)Cc2cccnc2O)c1 c1(C(=O)NCC2C3CN(C(c4cc(Cl)c[nH]4)=O)CC23)ccc(F)cc1OC(F)F C(=O)(CC(C)C(F)F)N1CC(NC(CCN(CC)CC)=O)C(C)C1 C1(NC(C2(C)CCCCO2)=O)CCOC2(CCN(C(=O)CSC(F)F)CC2)C1 c1(OC)ccc(NC(=O)C(F)(F)F)cc1C(c1ccccc1)C1CC1 C1(CNC(CN(CCC)C)=O)C(C)CCCN1C(=O)CCc1ccnc(Cl)c1 Cc1ccc2c(=O)c(C(=O)NC3(CNC(=O)C#CC4CCCOC4)CC3)c[nH]c2c1 N#Cc1cc(C(N2CC(NC(c3cnc(-c4cccnc4)s3)=O)C3CC23)=O)no1 Cc1cncc(C(=O)NC2CCCC2NC(=O)C(O)CCN(C)C)c1C C1(c2ccccc2)(NC(N(C(C2CCCC2)C)C2CC2)=O)CC1(C)C N1(C(C(COC)C)=O)CCC(C)(C)C1CC(=O)Nc1ccc(Cl)c(OC)c1 c1(C(=O)NCC2(O)CN(C(C(C)SC(F)(F)F)=O)C2)ccc2c(c1)C=CCC2 C1(C(=O)NC(c2ccccn2)C)CC2(C1)CN(C(c1ccc(Cl)c(Cl)n1)=O)C2 C1(C(N2CC(NC(CN(CC)CC)=O)C2)=O)COC(C(F)(F)F)C1 C1(C2CCCN(C(C3CC4C=CC3C4)=O)C2)(NC(c2c(C)nsc2C)=O)CC1 c1(CC(=O)NCC2(NC(C3C(C=C)C3)=O)CCCC2)ccccc1SC c1(C(=O)NC2C(CNC(C(C)(C)c3cc[nH]n3)=O)CCC2)cccc2ccnn12 C#CC1CN(C(=O)CSCC)CCN1Cc1ccc(F)cc1F N1(C(C(C(CC)C)C)=O)CCC2(C1)CN(C(=O)CCc1cn(C)nn1)CC(C)O2 N1(C(=O)C(F)C2CCC2)CCCN(C(c2ccccc2)=O)C(CO)C1 C(C(Cc1ccccc1)CC(C)C)NC(=O)OC.C12CN(CC1(F)F)C2=O Cc1cnccc1C=CC(=O)NCC1CCC1NC(=O)C(c1cccnc1)O C1(NC(C(C)(C)c2cnsc2)=O)CC2CCC(C1F)N2C(c1cncnc1)=O C(=O)(CCCN(C)N=O)N1CCCC(C(C)NC(C(CNC(C)=O)(C)C)=O)C1 C1(NC(c2cnc(Cl)s2)=O)CCOCC1NC(C1CC12CC2)=O c1(OCC)ccc(C(=O)N(CC(C)NC(c2c(Cl)cncc2Cl)=O)C)cc1O N1(C(CCCN(C)N=O)=O)CCN(C(c2c[nH]c(=N)s2)=O)C2CCCCC12 CC(C)(O)C(F)C(=O)N1CCC(O)CC1C(=O)NOCC(F)(F)F C(=O)(C(C)(C)C(F)F)N1CCCC(CN(C(c2cc(C(N)=O)[nH]n2)=O)CC)C1 C1(CC)CCC(C)N1C(c1cccnn1)C(=O)NC(C)CC c1(N(CC(=O)NC(CNC(Cc2c(C)occ2)=O)CO)C)cccc(C#N)c1 c1(C(=O)NCC(CC)NC(=O)COC2CC=CC2)c(N)cc(C)cc1F c1(C(N2CC(F)(C(C)NC(C3(C4CCCCO4)CC3)=O)C2)=O)cc(N)ccc1Cl C(=O)(CC1=CCOCC1)N1C(C(=O)NC(c2nc[nH]n2)C)CN(C)CC1 C1(CC(=O)OC)CC2(CCN(C(c3cnc(S)n3C)=O)C2)C1 CC(C(=O)NCC(F)CNC(=O)Cc1ccc(CO)cc1)C(F)(F)C(F)F C12(NC(c3ccc(CC(C)C)cc3)=O)CCOCC1CN(C(c1cnns1)=O)C2 N1(C(c2c(=N)[nH][nH]c2)=O)Cc2nccn2CC(NC(C2COCCO2)=O)C1 C(=O)(CCC(F)(F)C(F)F)NC1C(CNC(COCCOC)=O)CCC1 c1(C(=O)NCC2CCCCN(C(C3(C4CC4)CC3)=O)C2)noc2cc(F)ccc12 C#Cc1cccc(C(N2CCCC2(C)C(=O)OC)C(=O)NCc2ccccc2)n1 C1(NC(CCSC)=O)C2CC3C1C3C2C(N1CC(F)(F)C1C1CC1)=O C(=O)(C(C)C(O)C(C)C)N1CCC(C2N(C(c3c(C)cn(C)n3)=O)CCC2)C1 CCC(C(=O)NC(C)C(C)NC(c1ccnc(C(F)(F)F)c1F)=O)C(C)(C)CC C12(NC(COC)=O)CCCN(C(C3CN(S(=O)(=O)CC)C3)=O)CC1C2 Cc1ncc(CNC(=O)C(C2CCCCC2)NC(=O)CC2CC2(C)C)s1 N1(C(c2nc(C)sc2C)=O)CC2CC(NC(c3cccc(CCO)c3)=O)C1C2 C1(c2n(C)ncc2)CN(C(=O)CCc2cc[nH]n2)CC1NC(c1ccsc1)=O CN1CCC(CCNC(C2CC=CCN2C(c2ccn(C)c2)=O)=O)CC1 CC1CN(C(c2ccc(-c3nn[nH]n3)cn2)=O)Cc2ccccc21 c1(C(=O)NC(C(C)(C)NC(C(CC)N2CCCC2=O)=O)C)ccc2snnc2c1 C1(C(=O)NCC2CC(NC(Cn3nc(C)c(Cl)c3)=O)C2)CCC(C(C)C)NC1=O C#CCCCC(=O)N1CCC(N2CCN(C(=O)CN(C3CCSC3)C)CC2)CC1 c1(OC)cccc(C)c1CNC1CCC(C(=O)NC(CO)C(C)C)C1 C(=O)(C1Cc2ccc(Cl)cc21)NCCC(C)NC(c1ccc(S(N)(=O)=O)nc1)=O C(=O)(CCC(C)(C)F)N1C(CNC(C2C(OC)CCC2)=O)C(C)CC1 C1(CC)CN(C(=O)CCCNC(N)=O)CCN1C(C1CC(=C(F)F)C1)=O N1(C(c2cnc(OCC)s2)=O)CCN(C(=O)CCn2cnnn2)C(CC(F)F)C1 N1(C(C(CC)(C)C(N)=O)=O)CCC(NC(=O)C=CCF)C(F)(F)CC1 N1(C(c2ccc(=O)n(C)c2)C(=O)NC)CCC2CCC(O)CC2C1 c1(C(=O)NC(C(CO)NC(C(CO)N(C)C)=O)C)nn(CC(F)(F)F)cc1Cl c1(C(=O)NC(C(C)C)CCN(C)C(C2CCC(F)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(CCCC(=O)N(C(C)CNC(c1cnc(CC(C)(C)C)o1)=O)C)NCCC c1(NC(C)Cc2nccn2C)nc(=NC2CC=CCCC2)[nH]c2ccsc12 c1(CC(=O)N(C2CCC(NC(c3cccs3)=O)C2)C)cc(C2CC2)on1 C1(C(=O)NC(CC=C)CNC(c2nc(C)no2)=O)CCc2nnc(O)cc2C1 N1(C(CCCCCCSC)=O)CCC2CCC(C1)N2C(c1ccc(C)s1)=O c1(C(=O)NCC2(C(C)(C)O)CN(C(C(COC)C)=O)C2)cnnc(C)c1C C1(NC(C(CC=C)C)=O)C2CC3C(C2)C13C(=O)N(C)C(c1cc(C)on1)C N1(C(C(C)=CC)=O)C2CCCC1CN(C(=O)C(COC)CC(C)C)C2 C1(CNC(C2(C)CC(=C)C2)=O)CCCCC1N1CCN(C(=O)C(F)C(C)C)CC1 C(=O)(C(CCO)NC(=O)NC1CC1)NC(C)CN(C)C(C1(C(F)F)CCCC1)=O C1(C(=O)NCC2CN(C(c3coc(Cl)n3)=O)CCO2)CCCCS1(=O)=O Cc1ncc(C(=O)NC2CC(C)N(C(=O)C=CC3CCOC3)C2)cc1N C(CCN=c1ccnc(NCC2CC(=O)N(CC)C2)[nH]1)N1CCC(CCOC)C1 C(=O)(C(C)(CC)C(=O)N1CCC(C)(Cc2cn(Cc3ccno3)nn2)C1)OCC C(=O)(C1=CC2(CCOC2)C1)NC1CCC(N(C(CCC2N(C)CCC2)=O)C)CC1 C(=O)(CS(C)(=O)=O)NCC(C1CCN(C(C2CCCN(CC(F)F)C2)=O)CC1)C C12CN(CC(F)(F)C1)CCN2.N1(C(c2ccc(Br)s2)C)CCC(O)CC1 c1(C(=O)NCc2cc(C(=O)NC(CC)C(C)C)n[nH]2)cccc(OC)c1 Cn1[nH]c(-c2nc(C(C)O)nn2-c2cccc(Cl)c2)nc1=O c1(NC(C2CC3CC(NC(=O)C(O)C(F)(F)F)C3C2)=O)cc2cccn2cn1 C=CCC(C)(CC)C(=O)NCCC1(O)CN(C(c2ccc(=N)[nH]n2)=O)C1 c1(C(=O)NCC(C)(CNC(=O)C(N)=O)OC)cnn(C(C)(C)C)c1N C(N=c1[nH]c(=NCC=CBr)c2sccc2[nH]1)C1CCC(=O)N1 C1(NC(C(C)N(C(=O)C2=CCCC2)C)=O)CCCC(C)(C)C1 c1(COCC(=O)N(CC(C)N(C(C=C(C)I)=O)C)C)ccccc1C CC1(C(N2CC(NC(c3cncs3)=O)C2)=O)CCCCC1(F)F COn1cnc(C)c1C(=O)NCC1(F)CCCN(C(=O)COCCN(C)C)C1 c1(OC)ccc(F)cc1NC(C1(COC)CCCN1C(=O)C1=C(Cl)CCC1)=O c1(OC)ccc(C(=O)N(CC(C)CNC(=O)CN2CCC(C)(C)C2)C)nc1Cl c1(C(=O)NCCC2CCCCN2C(C2COCCO2)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(Cc2cc(OCC)no2)=O)CCC(NC(C2(C)CCCN(C)C2)=O)C(C)C1 N1(C(COCC(C)C)=O)CCCC(CNC(=O)Cc2cncnc2O)CC1 Cc1coc(C(N2CCCC2CNC(C2CCOC2(C)C)=O)=O)c1C N1(C(c2c(SC)cn(C)n2)=O)CCC(F)(F)C(CNC(c2ncsc2C)=O)C1 S(=O)(=O)(CCCN)NC(C)(C)C.C123CC(CC1CNC(=O)N2)C3 CC1OCCC1CC(=O)NCCn1cnc(C(=O)NCc2cnc[nH]2)c1 C12(NC(c3ccc(CCC)s3)=O)CCCCCC1N(C(C1CCCCS1)=O)CC2 c1(C(=O)NC2C3CN(C(C(n4cc(C)nc4)(C)C)=O)C2CC3)nccn2nccc12 CC1CN(C(=O)CSc2cccc[n+]2[O-])CC1CCNC(c1ncn(C)n1)=O O=C(CS(=O)(=O)C1CCCC1)NCC(CNC(c1cccc2ncnn12)=O)CO C1(C(N2CCC(c3ccc(Br)cc3)C2)=O)CC(O)CN1C(c1cc(Cl)c(Cl)s1)=O c1(CC)c(C(N2CCC2CNC(C2C(Cl)(Cl)C23CC3)=O)=O)cnn1CC c1(C(C)NC(C(C)OC)=O)ccccc1-n1cc(CN2CCSCC2)nn1 O=C1NC2(CCO1)CN(C(=O)CC1CCCCN1C(C13CSCC1C3)=O)C2 N1(C(CN(CC)CC)=O)CC2(CCC(NC(C34CCCCC3C4(F)F)=O)CC2)C1 C1(C(C)C)CN(C(=O)CC(CC2CC2)NC(=O)CC2C=CS(=O)(=O)C2)CCO1 c1(CCC)cccc(CNC(=O)CS(C)(=O)=O)c1.C12CCC(C1)NC2=O C1(CCOC)CN(C(=O)CSCC(N)=O)CCN1C(=O)CC1(C(F)(F)F)CC1 C1(C)(CCNC(c2cc(CC)no2)=O)CCN(C(=O)CCC(=O)NC2CCC2)C1 c1(OCCOC)ccc2c(c1)CCN(C(=O)C(N1CCc3ccccc31)=O)C2 C1(C(=O)NCCCC2CCN(C(c3nc(C)n(C)n3)=O)CC2)CCC12CCCO2 N1(C(CCCOC)=O)CC2C(C(=O)NCC(C)(C)C3CC3)C2C1 C1(O)(C(C)NC(C(C)NC(=O)OC)=O)CN(C(=O)CC2CCCO2)C1 c1(NC(C(N2CCCC(COC)C2)C2CC3CCC3C2)=O)cc(C)ccc1C C1(C(N2C(C)CC(NC(C3(CCC=C)CC3)=O)C2)=O)CCC(C)=C(C)C1 C1(CNC(C(C)(C)CO)=O)CCN(C(c2ncc(F)cc2F)=O)C1(C)C CC1(CC2CC2)CCCS1.C1(CC(C2CC(OCC(=O)N)C2)=O)CCC(OC)C1 N1(C(C2(n3cc(Cc4cc(F)ncc4F)cn3)CCOCC2)=O)CC2OC(=O)OC2C1 c1(NC=O)ccc(F)c(Cl)c1Cl.CC(C)CC(C)(CC)O c1(C(=O)NCC(C)NC(=O)CCC2(C)CC2)ccc2c(c1)NS(=O)(=O)C2 CC1=CC(C(=O)NC(C(=O)NCc2ncnn2C2CC2)c2ccco2)SC1 N1(C(C(C)(C2CC2)OC)=O)CCN(C(c2ccc(CO)s2)=O)C(C2CC2)C1 C1(NC(c2cccc(N3CCCC3=O)c2)=O)(CO)CCN(C(c2ccoc2)=O)C1 C(CCCCCC(=O)NCc1cc(C2CC2)on1)NC(c1nn(CC)nc1C)=O c1(C(N(CC(C)(C)CNC(=O)C(C)NC(C)=O)CC)=O)ccc(C)cc1SC C#CC1CCC(NCc2ncc[nH]2)C1.c12ccc(cc1)CO2 Cc1nc(C(N2CC(c3cccc(F)c3)CC2C)C(=O)NC2CCC2)sc1C Cc1ccc(OCC(=O)NC2CCCN(C(C3CC3C(F)(F)F)=O)C2)cc1 N1(C(C(C(=C)C)(C)O)=O)CC(C)(C)CCC1CNC(c1ccc(Br)cn1)=O N1(CCO)CCOC(C)(C(=O)NC2C3CCCCCC23)C1.C(C)(C)(C)N(CC)CC C1(NC(C(C)(C)NC(=O)OC)=O)CCCC(NC(=O)CN(C)S(N)(=O)=O)C1 c1(CNC(C(C2CCOC2)OC)=O)ccccc1CNC(=O)Cc1n[nH]c(C)n1 C1(C(C(=O)OC)C)CCN(C(=O)C(F)=CCCF)C1.C1(=O)CO1 O=C(c1nn(CCO)c(=O)[nH]1)NC1CC(F)C1 N1(C(C(C)NC(C2CCCC2)=O)=O)CC=CCC2(CCCC2)C1 c1(CN2CC(CNC(c3ccc(Br)s3)=O)C2)cnc(O)nc1O c1(C(N2CCC(CCNC(C=CCC)=O)C2)=O)cc(Br)c(O)nc1C C1(CNC(CNC(=O)OCC)=O)CCCN(C(=O)CC2C=CCCC2)C1 C1(CNC(c2nccc(C#C)c2)=O)CN(C(c2conc2C)=O)CC(C)(C)C1 c1(CNC(COC(COCC#C)=O)=O)nnc2nc(C)cc(C)n12 C(c1ccc(OCC)cc1)=CC(=O)NCCC(CNC(C(C(C)C)SCC)=O)O C1(CN(C(CC2C(NC(COCC(=C)C)=O)C2)=O)C)CC1(F)F N1(C(CC2(C=C)CC2)=O)CCC2CN(C(c3cc4ccsc4n3C)=O)CC2C1 C1(CC(=O)N(CC#C)C(C)C)(N(C)C)COC1 c1(C(CC)OC)ccc(OC)cc1.c1(C(C(=O)OC)NC)ccccc1 c1(C(=O)NC(C)CN(C)C(c2cncn2C)=O)ccc2c(c1F)CCC2 CC1(C(N2CCC(C(N)=O)C2)=O)C=CCN1C(C1CC2(CCC2)C1)=O C(C(C)(C)CC(=O)NC(CC1CC1)CO)NC(c1n(CC)ccn1)=O c1(C(N2C(C)CC(NC(C3(CO)CCCC3)=O)C2)=O)ccc(Cl)c(F)c1 c1(C(c2n(C)nnn2)NCCF)cccc(Cl)c1 c1(NC(CC(=O)N(C(C)C(C)(C)C(=O)NC2CC2)C)=O)ccc(O)c(=O)cc1 S(=O)(=O)(c1cnn[nH]1)n1c2nnc1n2CCOC.c1(OC)ccc(C)cc1C N1(C(CC2(C)CC2)=O)CC23CCCC2(C1)CN(C(=O)CC1CCCC(=O)N1)C3 C=CCC(CC(C)C)C(=O)N1CCC(n2cc(NC(=O)C(C)CC=CC)cn2)C1 CCC(CC(=O)NC1CCN(C(=O)Cn2ncn(C)c2=O)CC1F)C(F)F c1(-c2cc(C(=O)NCc3ccccc3F)ncc2)cc(F)c(F)c(F)c1F N1(C(CN(C(C)=O)C)=O)CC2CCC(CNC(=O)Cc3cn(C)cn3)C2C1 N1(C(Cn2c(C)ncc2[N+](=O)[O-])=O)CCCC2C1CCN2C(=O)Cc1cnsc1 C1(C(=O)NC2(COC)CCC2)CN(C(=O)C(C(C)C)NC(C)=O)CCO1 C1(OCC)CN(C(=O)CC2(NC(=O)CC3COCCN3C)CC2)CC1C(=O)OC Cc1cc(C(=O)NCC(O)CNC(=O)C(C)(F)F)cc(F)c1C C(N=c1[nH]cnc2ccc([N+](=O)[O-])cc12)C1C2CN(C(c3cc(Br)n[nH]3)=O)CC21 N1(C(CCCC(=O)N(CC)CC)=O)CC(NC(=O)C(O)C(C)C)C2CCCCC12 C1(C(N2CCC(C(N(CCOC)Cc3ccc(Cl)cc3)=O)C2)=O)C2CCN1CC2 c1(C(N2C(CCNC(=O)C=C(C)Cl)CC(OC)C2)=O)ccc(C)c2ncccc12 Cc1cn(CC(=O)NC(C)CCN(C)C(c2cn[nH]c2)=O)c2ccccc12 CC1CN(C(c2ccc(CC3CC3)o2)=O)CCC1NC(=O)CCc1cnoc1 C1(C(N2CC(CCNC(c3n[nH]c(CO)n3)=O)C2)=O)CC=CCC1 c1(NC(C(C2CCN(CCc3c(O)n[nH]c3C)C2)C)=O)ccc(F)nc1F O=C(C1=C(Cl)CCC1)NCC1CCCCN(C(C2CC(O)CN2C(N)=O)=O)C1 c1(CCC)cc(=NC(=O)CC(C)n2ccnc2)[nH][nH]1 c1(C(=O)NC2C(NC(CSc3n(C)nnn3)=O)COC2)cncc(NC2CC2)c1 C1(NC(c2ccc(CC)cn2)=O)CC(F)CN(C(=O)CCOCC2CCCO2)C1 C1(CNC(Cc2cc(C)ns2)=O)CC2(CO1)CN(C(=O)C=C(Cl)Cl)C2 C1(CC(C)NC(c2ccc(O)nc2)=O)CCN(C(C2(C(F)F)CCCO2)=O)CC1 C1(CNC(C(C2CCOCC2)C)=O)CN(C)CCN1C(c1cnc2n1CCC2)=O Cc1ccc(F)c(C(=O)NC2CCOC2C(=O)NCC2(CO)CC23CCC3)c1 N1(C(c2cc(CC)on2)=O)CCCC(CNC(c2ccsc2CN)=O)C1 c1(C(N2C(C)C(NC(=O)CC3CCOC3)CC2)=O)ccc2c(c1)CC2 Nc1ccc(C(=O)NCCC2CCCN(C(=O)CC3CNC(=O)C3)C2)cc1F c1(CCC(=O)NNC2=NCC2)nnc2n1CCNC2 c1(C(=O)NCCCNC(CCOCCC)=O)ccc2c(c1)CC(C)(C)O2 c1(C(=O)NCC2C(C)CN(C(=O)C(C)SC(F)(F)F)C2)cc2ccoc2cc1F C(C1c2ccccc2CC1C)NCc1cc(OC)cc(Cl)n1 C12(C(N3CC=C(C)CC3)=O)CCC(CN(C(c3cnn(CCO)c3)=O)C1)C2 N1(C(CC(CC)OC)=O)CCN(C(c2cn(CCF)nn2)=O)C(CC)C1 CC#CCC(CO)NC(C1CCC(C2CC2)N1C(c1cnn(C(F)F)c1)=O)=O c1(NC(C2N(C(C(CCCC)O)=O)CC(O)C2)=O)ccnc(S(C)(=O)=O)c1 CCC(C)(CCC(C)C)C(=O)NC1CCN(C(C2CCCCS2(=O)=O)=O)CC1C C1(C2CCN(C(C3CC3[N+](=O)[O-])=O)C2)(NC(=O)C=CC2CCCCCC2)CC1 N1(C(c2c(OC)ncnc2C)=O)CCN(C(=O)Cc2c(C)noc2C)CC12CC2 Cc1ccc(C(=O)NCC=CCNC(=O)CC(C)N(C)C)c(F)c1C C1(c2n(CC=C)nnn2)(N(Cc2nnc(COC)o2)CC)CCCCC1OC c1(N(CCC=C)CCC#N)ccc(S(=O)(=O)NC(C)CO)cn1 C1(NC(=O)C2CC2)CCOC12CCN(C(C1CCCOC1c1ncc[nH]1)=O)CC2 N1(c2sc(C#N)c(Cl)n2)Cc2ccccc2C(CNC(c2cnc(Cl)cn2)=O)C1 Cc1cnc(CCNC)c(C)c1.C12CN(C(=O)OC(C)(C)C)CCC1CCN2 N1(C(C2CCCC(NC(C3C(C(C)C)OCC3)=O)CC2)=O)CCC2CC1C(=O)O2 C1(C(=O)NC(C2OCCN(C(c3ncc(OC)cn3)=O)C2)C)CNC(=O)CC1C C(CN(C(=O)C=CCN1CCCC1)C)(CO)(CO)NC(CC(C)NC(N)=O)=O c1(NC(CNC(CCOC)=O)=O)cccc(NC(C2(C)CCC(C)C2)=O)c1 Nc1cc(Cl)nnc1C(N1CCC(O)(CNC(c2c[nH]nc2C2CCC2)=O)C1)=O C(=O)(C(C)(C)C(=O)NC1(CNC(=O)NC2CC(F)(F)C2)CCC1)N(C)C c1(C(N2C(CCc3cn(C(C)CO)nn3)CCC2)=O)ccc(Cl)c(Cl)c1 c1(OCC2(O)CN(C(C3(C(=O)NC)CC3)=O)C2)cc(C(=O)N(C)C)cc(F)c1 Cc1ccc2c(c1)CC(C(N1CCN(C(C3CC4CCC4C3)=O)CC1)=O)S2 CC1CN(C(=O)CN2CCC2)CCC1NC(=O)C(C)(CN(C)C)c1ccccc1 c1(CNC(C2(CCNC(C3CCCSC3)=O)CCC2)=O)ccc(CO)o1 N1(C(C2CC(C)OC2)=O)Cc2nccn2CC(NC(C23CCCC(C2)OC3)=O)C1 c1(CN2C(CC(=O)NC(=O)NC)CCC2)ccc(CO)c(C(C)(C)C)c1 CCC(C)CC(=O)C(=O)N(C1CN(C(=O)C(C)CN(C)C)CC1(C)C)C C(=O)(C(F)C(C)(C)O)NC(C)(C)CCCNC(c1coc(C(F)F)c1)=O n1(COC)ccc(C(N2CC(C(N)=O)(CNC(=O)CCc3ccsc3)C2)=O)n1 C(CC1=CCN(C(=O)CC2=CCCCC2)CC1)NC(C1CC2(CC(=C)C2)C1)=O c1(OCC)cccc(C2CC2)c1.n12nccc1C(C)N2 c1(CCC(=O)NC(c2c(OC)ccc(C)c2)C)nc2ccccc2o1 N1(CCCCC)CCCC1NC(=O)NCCC1CCCN1C Cc1c(NC(c2c(-c3ccc(C(C)(F)F)cc3)cnn2C)=O)cc(F)cc1Br c1(C(N(CCCCNC(C(CC)c2cccnc2)=O)C)=O)ncnc(O)c1Cl C1(C(N(CC(=O)N(CCC(=O)NC)C)CC)=O)CC(=O)N(OC)C1 c1(C(N2CCCC(C)(CC)C2)C(=O)NC2CCOCC2)c(Br)cc(OC)cc1Br N1(C(CCC#C)=O)CC(NC(=O)CCNC(c2ccc(F)cc2)=O)C(F)C1 N1(C(c2c(CC)cno2)=O)CCOC(CCNC(c2cscn2)=O)C1 CC1(C)CN(C(C2(C)CC2c2ccccc2)=O)CC1NC(C1(CCF)CC1)=O C(=O)(C1OCCc2cc(O)ccc21)NCC1CCN(C(c2cc(C#N)on2)=O)C1 CCC(F)(F)CCn1nc(-c2ccc(C(F)(F)F)cc2)nc1C(C)OC CC(Cc1cnn(C)c1)C(=O)NCCN(C(C1(N(C)C)CCCC1)=O)C1CC1 N1(c2snc(C(=O)OCC)n2)CCC=C(C(=O)N(C)CC2CCOC2)C1 c1(CC(=O)NC2C3(CC(NC(CC4CCN(C)CC4)=O)C3)C2)ccc(Cl)c(Cl)c1 C(CC(C)(C)C(=O)NC1CCN(C)C(C(C)C)C1)NC(C1C(OC)CCC1)=O O=C(C1COc2ccccc21)N1CCN(C(c2n[nH]cc2F)=O)C(CCO)C1 C(=O)(C(C)(C)CCCNC(c1cnc(C)n1C)=O)NC(CC)C(O)C(C)C N1(C(c2ccc(OC)cc2)C(=O)NCC=C)CCN(CC)CC1 N1(C(=O)C(C2CCOCC2)F)CCC(F)(C(N2CCC(F)(F)C2)=O)C1 c1(CCNC(=NCC=C)NCCC2(C)CC2(F)Cl)ccc2c(c1)OCCO2 c1(C(N(CC(O)CNC(c2ccccn2)=O)C)=O)sccc1S(C)(=O)=O c1(NC(N(C2C(CC)CCC2)C)=O)ccc(OCC#N)cc1 C(=O)(C1=C(C)OCCS1)N1CCC2C(NC(c3nn(CC)c(O)c3)=O)C2C1 N1(C(C(CNC(c2cn(C)nn2)=O)O)=O)CCC2(CC1)CC2 NS(=O)(=O)c1ccc(NCCOCCF)cc1Br C1(OCC(=O)NC(C(=O)NCc2ccoc2)C2CCCO2)CC=CC1 c1(CNC2(c3nnnn3CC)C(CC)COCC2)cccc(F)c1OC(F)F C1(C(C)C)CN(C(=O)CC2CCC=CCC2)CCCN1C(=O)C(CO)NC(N)=O Cc1ccc2cc(C(N3CCN(C(=O)C4=COCCO4)C(C)C3C)=O)ccc2n1 c1(C(N2C(CNC(=O)C(C)(O)C3CCC3)CC(C)(C)C2)=O)ccc(N)c(F)c1F C1(O)(CCNC(c2c(C)noc2C)=O)CCCN(C(=O)CCCOC(C)(C)C)C1 C(=O)(CC(C)C(F)(F)F)N1CCC(C)(NC(CC(CCC)C)=O)C1 CCC(C)C(C)C(=O)NC1(CCNC(C2(Cl)CC2)=O)CCC1 c1(C(=O)NC(C=CC(=O)NC2C(OC)C(O)C2)(C)C)nc(=N)cc[nH]1 c1(OC)cc(F)c(F)cc1NC(=O)C(c1ccc(Br)cc1)C C(CC(=O)N1CCCCC1CNC(=O)C1=CSCS1)(C(F)(F)F)N(C)C C1(CNC(C2CC=CCO2)=O)CN(C(c2sccc2F)=O)C2CCCC2O1 Cc1cccc2c1CN(C(C1(CO)CCN(C(=O)COCCN(C)C)C1)=O)C2 c1(C(=O)NC2CCN(C(c3c(C)nsc3C)=O)C(C)C2)c(F)ccc2occc12 C12(NC(CCCC#C)=O)CCCC1N(C(=O)CCF)CCC2 O=S(=O)(C1CCC2(CC2)C1)N1CCC(CN2CCCC2)CC1 CS(=O)(=O)c1ccc2[nH]cc(CN3CCCC(C(N4CCNC(=O)C4)=O)C3)c2c1 c1(C(=O)NC2CCN(C(C3C(C)C3C)=O)C2)cccc(Cl)c1O CCC(Cc1ccccc1C)C(=O)NCc1cc(C#N)cs1 Cc1cc(-c2cn(Cc3cccc(NC(=O)CCOCCOC)c3)nn2)cc(Cl)n1 c1(C(=O)NC(C)CN(C)C(C2CCCCS2(=O)=O)=O)cn(C)c2ccc(F)cc12 c1(OC)cccc(Cl)c1C(=O)NCCCCNC(C1CCCC(C#N)C1)=O C1(CNC(CCC2(C)CC2)=O)CN(C(c2cncc([N+](=O)[O-])c2)=O)C2(CCC2)C1 C1(CC(=O)NCCCN(C)C(c2csc(C3CC3)n2)=O)CCCS1(=O)=O CN=C(NCC(c1ccsc1)C)NCC(C)(O)Cn1cc(Br)cn1 c1(C(c2nnnn2CC(F)F)NC(C)Cn2cccn2)nsc(COC)n1 CCC(C)C(C(=O)NCCCNC(=O)CCF)NC(C1(C)CC=CCC1)=O C(C)(CCC(=O)N(C1CCN(C(C2CC2F)=O)CC1)CCO)OCC C(CCC(C)C)=CC(=O)NC(C(=O)NC(C#C)C1CCC1)C1(C)CC1 c1(C(=O)NC(CCN(C(C=CC=CC)=O)C)C)ccc2ccn(C(C)(C)C)c2c1 c1(-c2cnc(CNC(c3c[nH]c4ncccc34)=O)nc2)cc(F)c(F)c(F)c1F CP(C)(=O)c1ccccc1C(=O)NCCCOCCNC(c1c[nH]c(=O)cn1)=O C1(CNC(C2CCC(CNC(C(C)SCC)=O)O2)=O)CCCCC1(C)C C1(CNC(C(c2cccc(O)c2)C)=O)CCCCN1C(=O)Cn1cccn1 c1(OC)cccc2[nH]nc(C(=O)NCC(O)CCNC(C3CCC(=O)C3)=O)c12 C1(CC)(CC)CC2N=CN=C(C3=C(N1)CSC3)N(CCC(C)OCCO)C2 C#Cc1ccccc1C(=O)NCC1CCCN1Cc1ccnn1-c1ccccc1 C1(NC(C2CCCC3CC23)=O)C=CCN(C(C2CCCO2)=O)C1 C1(F)(CNC(CCSCC(C)C)=O)CCN(C(=O)CC2(n3ccnn3)CC2)C1 C1(CC)(CNC(=O)C(CO)NC(=O)C(C)c2ccco2)CCCC1 C(CNC(c1ccc(F)o1)=O)(C(C)(C)C)NC(c1c(CCC)[nH]cc1)=O c1(C(N(C2C3CN(C(C4CCS4(=O)=O)=O)CC23)C)=O)cc2n(n1)CC(C)(C)CO2 N1(CC(=O)OCC2(N3CCOCC3)CCCOC2)CCOc2ccc(Cl)cc2C1 CC1(C(=O)NCCc2ccnc(F)c2)CCN(C(c2ccccc2)=O)C1 C=CC1(C(=O)NC2CC3(CCC3)C2O)CCN(C(=O)CCOCC(C)C)C1 c1(CCNC(N2CCC(C)(c3onc(CC)n3)C2)=O)cccc(C)c1F C(CN=C(NC(c1cccc(Br)c1)C)NC1CCOC1)c1c(OC)nsc1 N#Cc1ccc(Cl)c(C(=O)NCC2CC(NC(c3ccc(C(F)F)nc3)=O)C2)c1 C1(C(CO)NC(N2CC3CC3C2)=O)CCC(F)(F)CC1 c1(C(=O)NCCC2(CNC(c3nnn(C)n3)=O)CC2)cc2ncccc2[nH]1 C(=O)(CCCC(C)(F)F)N1CC2(CN(C(C(=Cc3ccncc3)C)=O)C2)C1 N1(C(C(C)Cc2ccc(F)cc2)=O)CC(C)(CNC(c2cc[nH]n2)=O)CC1(C)C c1(C(=O)NCc2ccccc2C(F)F)cccc(C(N2CC(O)C2)=O)c1 N1(C(C2C(C3CN(C(C4(OCC)CCOC4)=O)C3)C2)=O)CC2CC=CCC2C1 N1(C(C(c2cccc(F)c2)C)=O)CC(NC(C2CC2(C)C)=O)CC12CCOCC2 C(=O)(C(C)(F)CC1CCCC1)N(C1CCN(C(c2cnn(C)c2N)=O)C1)C C1(NC(CCc2nccc(C)c2)=O)C2CCC(C2)C1C(=O)NCc1cn(C)cn1 C(=O)(C(C)CC(F)(F)F)NCCCNC(c1nc(COC)oc1)=O Cn1cc([N+](=O)[O-])cc1C(=O)NCC12CCC1CN(C(C1(C#N)CCOC1)=O)C2 C1(CNC(C(C)C)=O)CN(C(c2ccn(C(C)C)n2)=O)CCCO1 C1(NC(CCC(=C)Cl)=O)CCC2(CC1)CC(NC(c1cc(C3CC3)n(C)n1)=O)C2 c1(Cn2cc(COCC)nn2)c(OCC2CC23CCNCC3)cccc1Cl C1(NC(=O)CS(=O)(=O)C2CC2)CCC2(CCN(C(c3csnn3)=O)C2)C1 C#Cc1cccc(NC(N2CC(O)CC2CC(=O)Nc2cn(C)nc2O)=O)c1 N1(C(C2CC(C)N(C)C2)=O)CCC(F)C(NC(c2ccnn(C)c2=O)=O)C1 c1(CC(=O)NC2C(CNC(CC3C(C)(C)COCC3)=O)C2)ccc(F)c(O)c1F c1(C(=O)NCC(C)N(C(c2n(CC)ncc2)=O)C)ccc(C)c(O)n1 C#Cc1cnn(C)c1C(=O)NC1CC2CC1N(C(=O)CCC1CCOC1)C2 c1(OC)ccc2c(c1)CCCN2C(=O)CSCc1nc(C(F)(F)F)cs1 CC1(CC(=O)NC2CCCC2CNC(C2CC2(Cl)Cl)=O)CC(C#N)C1 C1(NC(CNC(C2C(C)C2)=O)=O)CN(C(=O)C=CC(=O)OC(C)(C)C)CC1(C)C CC1CN(C(c2cccc(CO)n2)=O)CC(CCNC(=O)CCCC2CC2)O1 c1(CC(=O)NCC)ccnc(N2CCC(OCCOC)C2)n1.C12CCOC(C1)C2 CCC(C)C(C(=O)NC1CC(NC(=O)C(C)Oc2ccccn2)C1)NC(C)=O C(=O)(CC(C=C)CC)N(C1CCN(C(=O)C(C2CC2)OC)CC1)CC#C Cc1ccc(CNC(=O)C(C2CCN(C(c3csc(C)c3C)=O)C2)C)cc1C S(=O)(=O)(c1cnc2ccccc2n1)NC1CCN(c2cc(C)nn2C)C1 CCC(C(=O)NC(C)(CNC(c1nc2cccnc2s1)=O)C(C)C)C(C)(F)F C1(NC(c2c(Cl)ccc(C)c2)=O)CC2(CCN(C(C3CCN(C)C3)=O)CC2)C1 N1(C(C=C(C)C(C)C)=O)CCN(C(C2CC2(Cl)Cl)=O)C(C(C)(C)C)C1 C1(CO)COCC2(CCN(Cc3ocnc3C(=O)O)C2)O1.c12cccc(c1)OC2 CCC(C)CC(C)C(=O)NC1CN(C(c2noc(-c3cccc(F)c3)n2)=O)CC1C C(=O)(C(C)C(O)C(C)C)N(C(CNC(C(COC(C)C)NC(C)=O)=O)C)C N#Cc1ccc(CN2CCN(C(=O)CCc3ccc[nH]3)CC2)c(F)c1F N1(CCNC2C(C)C2)C(=O)CN(CC(N2CCCCC2)=O)C1=O N1(C(c2c(C)nco2)=O)CCCC(C2CN(C(c3cn4c(n3)CCC4)=O)C2)C1 c1(CC(=O)NC2(C)CCN(C(CCCC=C)=O)C2)cn2c(C)cncc2n1 C1(CNC(C(CCC)OCC)=O)CC2COCC2N1C(C1COC(=O)N1C)=O c1(C(=O)NC(C(C)C)CNC(=O)C2CC2)cc2c(cc1F)OCC(=O)N2 C(CC(C)(C)CC(=O)NCC1(N(C(CC2(N(C)C)CC2)=O)C2CC2)CC1)OC N1(CC(=O)NCCCN(C(=O)COCCF)CC)CCCC1CO C1(C(N(C(CO)CO)CC)=O)CCOC(CNC(=O)CC2CC3CC3C2)C1 Cc1c(C(=O)NC(C)(C)CCNC(=O)CC2OCCCO2)noc1C1CC1 c1(C(=O)OC)cccc(CC(=O)NC2CCC(CCNC(=O)C(C)N(C)C)C2)c1 O=C1CCC(CC(N2CCC(N(C(=O)C(=O)Nc3ncc[nH]3)CCO)C2)=O)N1 C1(NC(C(COC)OC)=O)CCC(CN(C(=O)CCc2ccc(F)cc2)C)CC1 c1(NC23CC(C)(C2)CS(=O)(=O)C3)ccn2ncc(S(N)(=O)=O)c2n1 c1(COC)cc(C(c2nnnn2C)NCC2CCOC2(C)C)ccc1Br C1(C)(C(N2CCC(C(C)C(=O)NCC3C4CCCC34)CC2)=O)CNC(=O)C1 c1(OC)nccc(Br)c1C(=O)NC1CCC1NC(=O)CS(C)(=O)=O c1(CCC(C)NC(=O)C(CNC(=O)CC(O)C2CCCC2)N(C)C)ccccc1 Cc1cccnc1CCC(=O)NCCN1CCN(C(C2(CF)COC2)=O)CC1 O=C(C1CCSc2ccccc21)NC12CCN(C(=O)CCCCC3CC3)CC1C2 C=CCCCCCCCC(=O)NCCC1(CNC(C2OCCC2C(C)C)=O)CC1 C1(C(N2C(C)CC(NC(=O)C(C)(C)CF)C2)=O)CC(C(=O)NC)=NO1 c1(C(N2CCC(C(C(=O)NCC3(OC)CC3)C)C2)=O)ccccc1C#N N1(C(C(C)CF)=O)CCCC(NC(=O)CC2C=CS(=O)(=O)C2)CC1 C(C(=O)N1CCCc2nncn21)NC(C(CC)n1ccnc1)=O c1(OC)cccc(C(F)F)c1C(=O)NCC1CC2CN(C(=O)CC(C)OC)CC12 Cc1c(C(N2CCCCC23CCSC3)C(=O)NC(C)C)sc2ccccc12 CC1CCC(C)C1NC(=O)C(c1cccnc1)NC(=O)COC1CCCC1 N1(C(c2[nH]cc(C)c(=O)c2)=O)CC2CN(C(=O)C(C)(C)CO)CC(F)(F)C2C1 N1(C(C=C(C)CNC(c2cnc(Cl)n2C)=O)=O)CC(CO)C1(C)C c1(C(N(CCN(C(c2cnc(C(C)C)n2C)=O)CC)CC)=O)cc(C)c(F)cn1 C1(CC)CN(C(c2c(C)noc2C(F)F)=O)CCN1C(C1CCS(=O)(=O)C1)=O N1(C(c2nc(SCCC(F)(F)F)oc2)=O)CC2(CCN(C(=O)COCC)CC2)C1 C12CCCCN1CC(C1CCCCC1)C2.C1(CC(=O)NC(C)=O)CCCCCC1 N1(C(C(C)SCCl)=O)CCN(OC(=O)NC2CC2)CCC1C C(=O)(C1OCCn2ccnc21)N1CCC(C)(NC(Cc2ccc(C)s2)=O)CC1 C12(C(=O)NCC(C3CC3)NC(c3c(N(C)C)cccc3)=O)CCC(CC1)OC2 C(=O)(C1=CCCC1C)N.C(CO)(C(=O)NC(C)C=CCCC(=O)OC)SC N1(C(c2c(C)ccnn2)=O)CCCC(C2CCN(C(=O)C3=CC(C)(C)C3)C2)C1 C1(NC(CC(CNC(CCNC(=O)C2CC2)=O)C2CCC2)=O)CCCC2(CCC2)C1 c1(C(c2nnnn2CCC(C(C(C=C)NOC)=O)=O)NCC)ccc(CC)cc1 C1(NC(C(C2CCCO2)OC)=O)CCN(C(=O)COCc2cccc(C)c2)CC1 c1(OC)cnc(C(=O)Nc2cccc(Oc3ccnc(C(F)F)c3)c2)c(OC)n1 c1(C(=O)NC(CCOC)CNC(C2(O)CCCC2)=O)cc(S(N)(=O)=O)cs1 c1(C2(C(N(CCN(CC(F)(F)F)C)C)=O)CC2)cccc2c1OCC2 O=C(CCCN1CCCC1)NCC1CC1CNC(c1sccc1C1CC1)=O C1(N(C(=O)C(F)C2CC2)C)CCN(C(c2csc(CC(F)(F)F)c2)=O)C1 C1(CNC(C(COCC)NC(=O)C(C2CCOCC2)=O)=O)CCC(F)(F)C1 N1(C2CCc3c(cnc(C)n3)C2)C(=O)C2CC3(CCCCCC3)CCN2C1=O c1(CNC(=O)Nc2ccc(OCCF)cc2)cccc(C(F)F)c1 c1(NCCC2CCC(NC(CSCC#C)=O)C2)ccc(-n2ccnc2)cn1 C1(NC(C(CCC2CC2)NC(c2cnncc2O)=O)=O)CCCC2(CCC2)C1 n1(NC(C(C(C)C)c2cn(CC(F)CCN(C)C)nn2)=O)cc(S(N)(=O)=O)cn1 C1(C)(CNC(c2onc(CC)c2C)=O)CCN(C(=O)CCCNS(C)(=O)=O)CC1 c1(C(N2CCC(CC=C)(NC(c3cc(Cl)ns3)=O)C2)=O)cc2n(n1)CCC2 C1(CC(=O)OC)CCCCC1N=c1cc(Cl)nc(C2CCC2)[nH]1 C1(NC(CCCOCC)=O)CCN(C(=O)CCn2nc(C)nc2C)CCC1(F)F c1(CC2CC(C(N(CCN(C)C(c3ccccc3)=O)C)=O)C2)ccccc1 N1(C(COC2(C)CCOCC2)=O)CC(F)(F)CC1(C)CNC(C1CCNC1=O)=O c1(C(N2CC(N3CCN(C(C4C=CCCC4)=O)CC3)C2)=O)ccc(OCF)cc1 Cc1nc2cc(C(N3CC=CC(NC(C4CC(=O)N4)=O)C3)=O)cnc2[nH]1 N1(C(CC)(C)C)CCC2(CCCN(CC3CCC(COC)OC3)C2)C1 CCC(CN1CCN(C2CCCN(C(=O)C(C)(C)C)C2)CC1)C(=O)O c1(C(N2C(CCNC(Cn3c(C)cnc3)=O)CCC2)=O)ccc2ccccc2n1 N1(C(C(C)SCCCC)=O)CCCC(O)(C(C)NC(=O)CN2CCCCC2)C1 Cc1cc(F)c(C(N2CCOCC2CNC(=O)CCc2scnc2C)=O)cc1F Cc1nc(C=CC(N2CCCCC(NC(=O)C=CC=C(Cl)Cl)C2)=O)[nH]c1C CC1C(C)N(C(=O)C=Cc2nccs2)CCN1C(c1ccc(Cl)cc1)=O N1(C(CC2CCN(C(C(CC(C)C)OC)=O)CC2)=O)CCC2(CC1)CC2C#N c1(C(=O)NC2CN(C(c3c(C)ncs3)=O)C2)cc2c(nc1O)CCCC2O CC1(C)CC(NC(c2ccc(N3CCCC3)cc2)=O)CN1C(C1C=CCC1)=O C1(CNC(CNC(C(c2cccnc2)C)=O)=O)CCCN(C)C1=O C(=O)(C(CO)C(C)(C)C)NCCC(=O)NCC(CCC=C)O N1(C(COc2cccc(OC)c2)=O)CC2(C1)CN(C(c1ccc(N)cc1C)=O)C2 N1(C(C2N(C)C(=O)OC2)=O)CCC2(CC(NC(c3csnn3)=O)C2)C1 CCC(C(=O)N1CC2(C1)CN(C(c1csc(CO)n1)=O)C2)C(C)C C1(C(=O)NCc2nc(Br)sc2Cl)Cc2ccccc2O1 c1(C(=O)NCCC(C)(C)NC(=O)COCP(C)(C)=O)ccc2ncccc2n1 C1(CNC(C(CC)NC(N)=O)=O)CCN(C(c2cc(C)ccc2N)=O)C(C)C1 C1(NC(C2(C=C)CCOCC2)=O)CCC2(CC1)CC2NC(=O)Cc1nc(=N)[nH][nH]1 Cc1ccc2nc(C(N3CCC(NC(=O)CCC(=O)NC(C)C)CC3)=O)cn2c1 C1(CNC(c2c(C)nc(COC)s2)=O)CN(C(C2COCCO2)=O)CC12CCC2 CCC(CCC(=O)NCC1CN(C(C2CC(C)(C)C2)=O)CC12CC2)OC C(CN=C(NCCC1SCCS1)NC1CC1)C1CC=CCO1 c1(C(N2CCC(N(C(C3(C#C)CCC3)=O)C)C(C)C2)=O)cc2cccc(F)c2s1 N1(C(CCCCN(C(C)C)C)=O)CCCCC1CNC(=O)CC(C)(C)O N1(C(C(C)N(C(C)=O)C)=O)CCCCC1C(=O)NC1(C)CC(C(N)=O)C1 N1(C(C(C=C)O)=O)CC(C(=O)N(CC(=O)NCC)C)C(CC)C1 c1(C(=O)NCCC(C)(C)NC(C(CC)c2cccnc2)=O)cnc(N)cn1 C12(CNC(=O)COC3CCCC3)CC(C1)C(NC(C1CCCC1(F)F)=O)CO2 C(=O)(C1=C(Cl)CCCC1)N1CC(CN(C(CCCN(C)C)=O)C)OCC1 C(CNC(c1ccncc1Cl)=O)(CC(F)(F)F)NC(c1cncc(N)n1)=O N1(S(CC)(=O)=O)CCCC1C(=O)N(C(C)CCNC(=O)C(F)n1cccn1)C N(C(=NCCc1cccc(Cl)c1)NC1CCSC1C)CC1(CSC)CC1 C(=O)(CC(CC)SC)NC(C(=O)NCc1cn(CCC)nn1)C O=C1CCCC(CC(=O)NC23CC(NC(c4cnccc4C(F)(F)F)=O)(C2)C3)N1 C1(C(N(CCCCC)CCO)=O)CCN(C(c2cc(C#N)[nH]c2C)=O)C12CC2 N1(C(C2CCC(=O)O2)=O)CCC2(CC1)CC2CNC(C1CCn2ncnc2C1)=O c1(CC(=O)NCC(C)N(C(CCCNC(=O)OC)=O)C)ccc(OC)c(F)c1 N1(C(c2oc(CC)c(C(=O)ON(C)C)n2)=O)CCCN(N2CCCCC2)CC1 C=CCC(C(=O)NCCOCCCCC)NC(=O)CN1CCCCCC1 N1(C(C2CCC(C)O2)=O)CCN(CCN(C(=O)CCc2cnn(C)n2)C)CC1 C1(C(N2C(CNC(Cc3c(C)ccs3)=O)CC2)=O)C2CC3C(C2=O)C13 c1(C(=O)NC2CCN(C(COC3(C)CCC3)=O)C2)ccc(C(C)(C)C)cc1N NC1CCc2cc(Cl)ccc21.n1(CCCSC)nnnc1C1(N)CC(C(N)=O)C1 c1(C(=O)NCC(CC)NC(c2c[nH]cc(F)c2=O)=O)ccc(Br)c(C)c1F C1(NC(C(CC)OC)=O)CCCCCN(C(c2c(C)nc(C3CC3)nc2C)=O)C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C2CC2)ccnc2[nH]cnc12 C1(CNC(C(C)Cc2ccccc2)=O)CN(C(C2(O)CCC2)=O)CC1(F)F N1(C(C(C=C)O)=O)CCCC(C(C)C(=O)Nc2cnn(C)c2CC)C1 C1(C(=O)NCC2C(C(=O)NC(CSC)(C)CO)CCCC2)CCCC(C#N)C1 N(C)(S(=O)(=O)N(C)C)CC(=O)NCC1(C)N(C(C=CCCC(C)C)=O)CCC1 Cc1c(C(N2CCC2CNC(=O)CC2CC2)=O)nnn1-c1ccccc1F c1(C(N2CCCC(CCNC(C3CCC3)=O)C2)=O)cn2cccnc2n1 CCCC(CNC(C1CCC(O)CC1)=O)C(=O)N(CC=Cc1ccccc1)CC CC(C)CS(=O)(=O)CC(=O)NC1CC(NC(c2cc(N)ccc2Cl)=O)C12CCC2 CNS(=O)(=O)NCC(=O)NC1CC(F)(CNC(=O)CN2CCCCC2)C1 C1(NC(c2cc(C)on2)=O)CC(C2CCN(C(=O)CC3CCC34CCC4)C2)C1 N1(C(=O)Cc2cnccn2)CC2CCCC(C1)N(C(=O)Cc1cccnc1O)C2 C1(C(=O)NC(CC)CN2CCCC2)CCCCN(C(=O)CCCC(C)C)C1 N1(C(C2N(CC)CC2)=O)CCC(c2ccccc2)(NC(=O)Cc2cnc[nH]2)C1 c1(CC)ncccc1C(=O)N(C(=O)C=CC1CC1)Cc1ccccc1.C12(COC1)CO2 C1(C(N2CCC(C(C)NC(c3ccn(CC)n3)=O)C2)=O)Cc2cc(C)ccc2S1 C1(C(=O)NCCN(CCCC)C)CC2CC2N1C(c1cccc(=O)o1)=O N1(C(CC2C(=O)NCC2)=O)C2CCC1CC(O)(CNC(C1(CO)CCC1)=O)C2 N1(C(=O)CSC(F)(F)F)CC(C2CN(C(c3cccc(F)c3Br)=O)C2)C1 C(=O)(CC(C(F)(F)F)OC)N1CC2C(NC(C3CCC(C(=O)OC)CC3)=O)C2C1 C12(NC(c3nc(OCC)oc3)=O)CCCCC1N(C(=O)CCC1CCC1)CC2 C1(C(=O)NCC2(NC(c3cn(C)nc3Cl)=O)CC2)CCCS(=O)(=O)C1 c1(C(=O)NC2(CCNC(C3CC(C#N)(OC)C3)=O)CCC2)cc2c(s1)CCCC2 N1(CCNC(C(C)Sc2ccccn2)=O)CCCN(C(c2cncs2)=O)CC1 CC12C3C4C1C1C2C3C41C(N1CCC(NC(C2CCCN2C2CCCC2)=O)C1)=O N1(C(CC=C)=O)CCCC(C2CCCN2C(=O)CCNC(=O)NCCC)C1 c1(-n2c(CS(=O)(=O)CCCC(C)CC(C)(C)C)nc(C)n2)cccc(S(C)(=O)=O)c1 Cc1cc(C(=O)NCC2=CCN(C(c3cc(C)nn3C3CC3)=O)CC2)cc(O)n1 N1(C(C(CCC)NC(=O)C=CC(=O)NCC2CC2)=O)CCCc2ccccc21 Cc1cc(Cl)c(C(=O)NCC2CCN2C(c2cocn2)=O)cc1C C1(NC(C(N(C(=O)CC2(C)CC2)C)C2CC2)=O)CC(C)(C)C1 c1(CCC)ccccc1C(N1CC(CNC(=O)CN(C(=O)C2CC2)CC)C(O)C1)=O C(=O)(C1=CS(=O)(=O)CCC1)NCC1(NC(C(C)OC)=O)CCCCCC1 C1(C(=O)NC2CC(C(C)NC(CCCOC)=O)C2)CCC(C)(C)C1 C12(C(=O)Nc3cc(C(=O)NC4CC4)no3)CCCC1CCC2 C=CCC(CC)C(=O)N1CC(F)CC1CC(=O)N(C)C(C1CN(C)CC1(C)C)=O c1(C(N2C(C(C)C)CN(C(C3CC3C(C)C)=O)CC2)=O)ccc2c(c1)CCN2C CCCC(C(=O)N1CCCC(N(C(=O)Cc2cccc(C(F)F)c2)C)C1)C(C)C C1(NC(C2CC(CC)N(C(C3C4CC5C(C4)C35)=O)CC2)=O)CCc2ncnn2C1 N#CC1CN(C(=O)CCC2CCCN2C(=O)CCCCN=[N+]=[N-])CCO1 c1(C(=O)NCCCNC(C2(CO)CC2)=O)ccc(-n2ccnc2)cn1 N1(C(C(C)CN(C)C)=O)CCC2(CCC2)C(NC(=O)Cc2cc(Cl)n(C)n2)C1 C1(C)(C(=O)NC2C(C)(C)C(C(N3CC(OCCF)C3)=O)C2)CC2CCC1C2 N1(C(C(=O)NCCOC)=O)CC(NC(=O)C=Cc2ccc(C3CC3)o2)CC(O)C1 c1(C(=O)NC2CN(c3nccc(OC)n3)CC2F)cc2c(C)c(C)ccc2[nH]1 O=C(C1=C2CCN=C2NC=C1)NCC1CCCSCC1 C1(C(N2C3CC(CN(C(C(CC(C)C)(F)F)=O)C3)C2)=O)CCC2COCCC2C1 CC1CCC(NC(=O)C=Cc2cn[nH]c2)CN1C(C1CC(=O)C12CCC2)=O c12ccc(cc1)OC(=O)N2.c1(OC)cnc(CNCC(C)N=[N+]=[N-])o1 Cc1ccc(CNC(C2COC(CNC(=O)C3=CC(C)(C)C3)C2)=O)c(O)n1 c1(CCC(=O)N(CCNC(c2cn(C)nn2)=O)CC)c(C)nc2ccnn2c1C N1(C(C2=CCC(C)CC2)=O)CC2CC(C)N(C(C3CCSC3)=O)C2C1 c1(C(=O)NC2C(CNC(=O)Cc3ccc(F)cn3)CCC2)cccc(Cl)c1O C1(CC(=O)NCCC(=O)NCc2n[nH]c(O)n2)CCCSC1 C1(CC(=O)NC2CCC(NC(c3c(NC)cncc3)=O)CC2)CCC(C)(C)CO1 c1(C(=O)NCCC(C)(C)NC(Cc2cnc(C)o2)=O)sc(=N)[nH]c1C Cc1cc(N)c(C(N2CC(NC(=O)Cc3cc(C(C)C)no3)C2)=O)c(F)c1 c1(C(=O)NC2CCC(N(C(=O)C=CC(F)F)C)C2)ncc(F)cc1F N1(CCN(C)C)CC(NC(=O)CCC(=O)NCc2ccccc2)CCC1=O N1(C(c2cccc(CCCSC)c2)=O)CCC2(CNC(=O)CO)CCCCC12 N1(C(C2(CCOC)CCC2)=O)CC2CCC1C(NC(=O)C(F)(F)CC1CC1)C2 C1(C(C(=O)NCC(CNC(C(C)CN(C)C)=O)c2cccs2)O)COC(C)(C)O1 C1(C(=O)O)(NC(C23CCC(C2)C3)=O)CC(O)C12CCC2 C1(C(=O)NC2CCC(NC(Cn3ccc(C)n3)=O)C2)CC(F)C(=O)N1 N1(C(C=C(C)C2CC2)=O)CCCC(C)(C(N2CCNC(=O)C2CCO)=O)C1 Cc1ccc(Br)c(CC(=O)NCC2COCCN2C(=O)C=CS(C)=O)c1 C(CC(C(=O)NOCC(O)COC)NC(=O)CC(O)CN(C)C)SC C1(NC(C2(C(C)C3CC3)CC2)=O)CC(CNC(=O)CN2CCCS2(=O)=O)C1(C)C Cc1csc(C(=O)NC2(C)CN(C(=O)CC3CCCC(C)C3)C2)c1Br c1(SCCC)cc(C(=O)N(CC(C)(C)NC(C2CC(C)C2)=O)C)ccn1 N1(CC(=O)NC(C)CC(=O)OC(C)(C)C)CCN(C)CC1C CC(C)C(CCN(C)C(C1(C)CCCCC1)=O)NC(=O)CCOCC1CC1 c1(C(N2CCC(N(C(=O)C=C3CCCC3)C)C2)=O)c(F)cccc1Br c1(SC)cc(C(=O)NCC2CCC2NC(C2(F)CCOC2)=O)ccc1[N+](=O)[O-] C1(C(=O)NC(CNC(c2cnn(CC)n2)=O)C)CCC(NC(N)=O)CC1 C1(C(CNC(C=COCC)=O)F)CCN(C(=O)CCC2CCCO2)CC1 C1(NC(COC(C)=O)=O)CCN(C(c2ccc(C(C)(F)F)c(Cl)c2)=O)CC1(C)C N1(C(C(CC)COC)=O)CCCC12CCN(C(c1ccc3c(c1)CCC3)=O)CC2 C1(CNC(CCC(C)(C)N(C)C)=O)CC2(CCC2)CN1C(c1ccoc1)=O CC(C)(O)C(F)C(=O)N1CCC(CO)(NC(c2ccnc(CO)c2)=O)C1 S(=O)(=O)(CC(=O)NC1CCCC(CNC(C2(C3CCCCO3)CC2)=O)C1)N(C)C C(=O)(C(C(C)C)C(C)C)NCCSCC(=O)NC(c1nc[nH]n1)CC c12cc(Cl)ccc1OC1(CC=C)CCN(C1)C2=O.C(=O)(C(C)CO)NCC1CC1 c1(OCCN(C)C)cccc(CN2CCC(NC(N3CCCCC3)=O)C2)n1 c1(C(=O)NCC(CNC(c2cccc(OC)c2)=O)O)c(Br)c(C)nn1C C1(NC(c2c(C)ccc(C)n2)=O)CC2CCC(C1C)N2C(C1CC=CCC1)=O N1(C(C2C(CC)C2)=O)CCC(NC(C2CSCC(=O)N2)=O)C(F)C1 C1(CNC(n2cc(NC(=O)CC3CCC3(F)F)nn2)=O)CN(C2CC2)CCO1.C1CC1 C(C1CCCCC1)=CC(=O)NCCN(CCOC)C(C1CC=CCO1)=O N1(C(C(C=C)(C)C)=O)CC(CNC(=O)C(N2CCOC(C)C2)=O)C(C)(C)C1 N1(C(C2CN(CC)C(=O)N2)=O)CCC2(CCCN2C(=O)CNC(=O)OC)C1 C(CC1CCOCC1)(C(=O)NCC=C(C)C)NC(CCC1CC(OC)C1)=O C(C(CC1CC1)C(=O)NCCN1CC(C)(O)C1)NC(C1N(CC)CC1)=O C(=O)(CC(C)(C)C(F)(F)F)NC1C(C)CCN(C(c2c(Cl)cn(CC)n2)=O)C1 c1(CN2CCC(CNC(=O)NC(CC(C)OC)C)CC2)ccc(Cl)c(F)c1 N1(C(c2ccc(CC)o2)=O)CCC(NC(=O)CC=C(C)C)C(CC)C1 CC(CCCNC(c1ccc(Br)o1)=O)NC(C1CC1c1ccccc1)=O c1(C(N2CC(CNC(C3CC(C4CC4)=NO3)=O)C2)=O)cc(Cl)ccc1C(F)F N1(C(CNC(=O)OC)=O)CCC(C2CCN(C(C3CCCC(=O)N3)=O)CC2)C1 N1(C(Cc2c(SC)cccc2)=O)CCN(C(c2ccnn2CCF)=O)CC1CF C1(C(=O)NC2CCC(n3cc(-c4n(C)ccc4)nn3)C2)C2CC3C(C2)C13 c1(CN2CCN(C(c3c(CC)nccc3)=O)C3C2C3)c[nH]c2cc(F)ccc12 N1(C(C2CCC(C)(F)CC2)=O)CCC2(CCN(C(=O)CCCC[N+](=O)[O-])C2)C1 c1(C(=O)NCC(CC)NC(=O)CCn2ccnc2)cn(C(C)C)nc1C C(=O)(CCCC(C)=O)NCCN(C(C(CC1CC1)OC)=O)C1CCCC1 c1(C(=O)NC2C(C)(C)C(CNC(=O)COc3ccon3)C2)ccc2cccnc2c1 c1(C(C(=O)NC(CNC(c2c(COC)ccs2)=O)C)N(C)C)ccccc1Cl c1(C(=O)NC2C(C(=O)NCc3ccc(C)c(C)c3)C2)ccc2c(Cl)ccnc2c1 c1(C(=O)NC(C2CN(C(C3CCCCCCC3)=O)C2)C)ccc2c(n1)CCCC2 c1(OC)ccc(NC(=O)C(=O)NC2CCCCC2N)c(F)c1 C1(C(NOCC(=O)OCC)=O)CC(NC(=O)CCC2(C#N)CCC2)C(O)C1 c1(C(=O)NC(CNC(C(CC)C(C)O)=O)C(C)C)coc(S(N)(=O)=O)c1 S(=O)(=O)(CC(=O)N1CCCC1C(C)(C)CNC(=O)C(c1ccc(C)s1)C)NCC C#CC1(O)CC(C(N2CCOC(CNC(=O)C=CSC)C2)=O)C1 C1(OC)CCCC1CC(=O)N(C)CC1CC1C.N12CCC1C2=O c1(OC)ccc(C(=O)NCC2(O)CCS(=O)(=O)CC2)c2ccccc12 N1(C(CCCc2n(C)cnn2)=O)CCC(CO)(CNC(C2(C)C=CCC2)=O)CC1 N12CCCC(C)(C)C1C2=O.C(=O)(CC(C)C(F)F)NCCNC(=O)OCC C(CCCC(=O)N1CC(C)(NC(=O)C(C)OCC(C)C)C1)OCC c1(C(c2nnnn2Cc2ccccc2)NC(c2cnc(Cl)s2)C)cn2ccnc2s1 C1(NC(C(C=C)O)=O)CCCCC1NC(C1(Cc2ccccc2F)CC1)=O CCCC(CCC)CC(=O)NC12CCC(C1)N(C(c1ccn(C)c(=O)c1)=O)C2 C1(C(N2CCN(C(C=CC=CC)=O)C(c3ncc[nH]3)C2)=O)CC2CCCCC2O1 C(C1OCc2ccccc21)NC(C1CCCN(C(C2CC3C=CC2C3)=O)CC1)=O CC1OC2CCC1(C(=O)NC1CC3(C1)CN(C(c1n[nH]c4c1CCC4)=O)C3)C2 N1(C(c2cc(C)c(Cl)cn2)=O)CCC2(CCCN(C(C3CCSC3)=O)C2)CC1 C1(NC(CCN(C(C(COC)OC)=O)C2CC2)=O)CCOCC1F C1(C)(CNC(C2(O)CN(C(C)=O)C2)=O)CSC(C)=N1.n12cc(nn1)NCC2 C(=O)(CC(C)(C)CNC(C1CCCCS1)=O)N1CC(SC)C1 C#CCCCCC(=O)N1CCCN(C(C)CNC(=O)Cc2cnsc2)CC1 N1(C(C2C(=C)C2)=O)CCN(C)C(CNC(c2cc(-c3cccs3)[nH]n2)=O)C1 N1(CCNC(C2CC2c2ccco2)=O)CCN(C(C2(N(C)C)CC2(C)C)=O)CC1 Cc1nc(C(N2CCOCC(CNC(c3n[nH]cc3Cl)=O)C2)=O)c2ccccn12 Cc1cc(C(=O)N(C2CCN(C(c3cn[nH]c3)=O)CC2)C)nc(O)n1 N1(C(=O)OC(C)(C)C)CCC2CCC12C(=O)NCc1cc(C(=O)O)on1 N1(C(c2ccc(C(C)C)cn2)=O)CCCCC(CNC(=O)Cn2ccnn2)C1 c1(C(N2CCC(O)(CNC(C(C#C)(C)C)=O)C2)=O)cc(C(N)=O)ccc1F N1(C(C(=O)NCC)=O)CCN(C(=O)CCCN2CCCCC2)CC1CF N1(C(C(CC)CC)=O)CC2(CCC2NC(c2nn(C)c(Br)c2C)=O)C1 Cc1c(C(=O)NC2CCN(C(c3csc(Cl)c3Cl)=O)CC2)ncn1C CCC(C(=O)NC1COCCN(C(c2conc2C)=O)C1)C(C)(F)F Cc1cc(=NC(C)c2cccc(C(F)(F)F)c2)[nH]c(N2CC3CC2CS(=O)C3)n1 C1C(F)(C(C)C)C(=O)N1.Cc1cccc(OC2CN(C(=O)OC(C)(C)C)C2)c1 N1(C(c2cccc(C#C)c2)C(=O)NCC(F)F)CCCN(C)CC1C C1(C=O)CC2CC1CC2(F)F.N12CCCN1C2.C12(CC1)C(=O)NC2C1CC1 C(=O)(C1=CCCC1C)NCC1CC(F)(CNC(C2(CC#C)CC=CCC2)=O)C1 C1(C)(NC(C(C2CCN(C(CCc3cc(C)[nH]n3)=O)C2)C)=O)CCN(C)C1 C(=O)(C1Cc2ccccc21)NCC(CC(C)C)C(=O)NCc1ccnc(Cl)c1 Cc1cc(F)cnc1C(=O)NC1CC1NC(=O)CCC1(C)CCC(=O)N1 C1(O)(C(=O)NCC(C)(CO)OC)CCOCC1.C1(=O)C(C2CCOC2)N1 C(C(C)(O)CC(=O)NC(CNC(=O)C(n1cc(C)cn1)C)C(C)(C)C)OC(C)=O N1(C(C(=O)NCC)=O)CC2CC(NC(C3(CC(=O)N(C)CC)CCCC3)=O)C1C2 C1(N(C(C(C)NS(CCC)(=O)=O)=O)C)CN(C(=O)CCCC(C)C)CCC1O N1(C(COc2c(C)occc2=O)=O)CCN(C(=O)COC2CCCC2)CC(O)C1 c1(C(N(CCCCNC(c2n(CC)ncc2)=O)C)=O)cccc2c1COC2 N1(C(Cc2c(C)non2)=O)CCCC(F)(CNC(C2C=CCCC2)=O)C1 C1(NC(c2n(CC)ccc2)=O)CCC(C)N(C(=O)CCCC#N)C1 Cc1nc2ccc(CN3CCC(C(=O)N(CC(c4nccs4)C)C)CC3)cc2o1 c1(C(=O)NC(C2CCN(C(CCC=C(C)C)=O)C2)C)[nH]cc2c1CCC2 c1(C(=O)NC2C(C(C)C)CN(C(c3ccns3)=O)CC2)ccc2c(n1)CCC2 C(=O)(CCCCNC(C1CCCC1)=O)NCC(CC)NC(=O)CC1CCCCO1 N#Cc1ccc(F)c(CN2CCC(CC(=O)NCc3nc(Cl)sc3Cl)C2)c1 C1(C(=O)NC(CC)CC(=O)N(C2CC2)CC23CCC(CC2)C3)CCCCC1(F)F c1(C(=O)NCC2(NC(C(F)=CC)=O)CC2)ccc(OC)c(C(F)F)c1 c1(CC(N2CCC(NC(c3c(C)ocn3)=O)C(C)C2)=O)cn2ccccc2n1 C(=O)(C(CCN(C)C)NC(c1c[nH]nc1C)=O)N1CC(O)(COC)C1 C1(C)(C(C(=O)NC2CCOC2)N(CCN(C)C)C2CC2)CCCC1 CS(=O)(=O)CC(=O)NCCCNC(=O)CN1CCC1CSc1cccc(Cl)c1 C(C(CC(F)(F)F)NC(=O)CCc1cnn(C)c1C)NC(C1(C)CC(=C)C1)=O c1(OC)nn(C)cc1C(=O)N(C)CC1(O)CCN(C(=O)CCNC(=O)CO)C1 c1(NC(c2n(CCSC)nnn2)c2cc(C3CC3)[nH]n2)cc(Br)ccc1[N+](=O)[O-] Cc1nn(C)c(C)c1C(N1CC=CC(NC(=O)C(C)n2cccn2)C1)=O N(C1CN(C(=O)CO)Cc2ccccc21)C(c1cn(C)nc1-c1ccccc1)=O C1(OC)CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)C(C)(C)CF c12ccc(cc1)c(=O)n(C)c2=O.c1(N)ccccc1F.N1(C=O)CCCC1CCO C(C(=O)NCC(C)C)(C(CC)C(C)C)N1CCC(C(CC)C(=O)NC(C)C)CC1 N1(C(CCCNC(C)=O)=O)CCC=C(CNC(C2CCC(=O)N(C)C2)=O)C1 C1(C(=O)NCC(=O)NC(CCNC(C(C)c2cncs2)=O)(C)C)CCS(=O)(=O)C1 N1(C(C(c2ccnn2C)C)=O)CCC=C(C(=O)N(C)C)C1.C12CC(C1(C)C)C(=O)N2 c1(CCCC)cc(N)c(C(=O)NC2CCCN(C(C3CC=CCC3)=O)C2)c(F)c1 C(=O)(CCC(=O)N1CC(OC)C1)O.N1(C(C)=O)CCC(C(C(=O)OC)CC)CC1 C(=O)(CCC(C)(F)F)C(CC1CCCN(C(CC(C)C2CCCC2)=O)C1)=O c1(C(=O)NC2CN(C(C=CC=CC)=O)CC2C)cccc2c1OCCCO2 C1(C(N2CCC(NC(C3(CCOC)CCC3)=O)C(C)C2)=O)Cc2cccnc2C1 C(=O)(C(C#N)C(C)(C)C)NC1C(NC(c2cc(CC)on2)=O)COC1 C(C(C)(C)C(=O)NC1CC(C)(C(=O)Nc2cncnc2C)C1)OCC C1(NC(c2c(COC)ncs2)=O)CCC12CN(C(=O)CSCCC(C)C)C2 C1(O)(C(=O)N(CCC(=O)NC(C)C)C2CC2)CN(C(=O)CCC2CCC(=O)N2)C1 c1(C(C)=O)cc(C(=O)NC2(C)CC(NC(=O)CCn3ccc(C)n3)C2)c(C)o1 c1(CN2CC(C(=O)O)(CNCC)C2)cc(OC)c2ccccc2c1 Cc1noc(C(=O)NCCN(CC(C)O)C(C2CCN(S(C)(=O)=O)C2)=O)c1C CC(C)C(C)CC(=O)N1CCC(n2cc(CNC(c3cccnc3O)=O)nn2)C1 c1(C(N2C(C)CCC(NC(c3ncc(F)cc3F)=O)C2)=O)cccc2c1CCN2 C1(COC)CN(C(=O)CC(C)C2CC2)CCN1C(C1(F)CCCCC1)=O CC(C)C(C(=O)NCCN(C)C(C1CCCN1Cc1ccsc1)=O)n1cncn1 N1(C(C(COCC)(C)C)=O)CCCCC(C(N2CCN(CC3CCC3)CC2)=O)C1 C1(C)(CNC(COCCOC)=O)CC(F)(F)CN1C(c1cc2ncccc2s1)=O N1(C(C2CSC2)=O)CCCC(C2CCCN(C(c3cc4occc4s3)=O)C2)C1 c1(C(N2CCC(NC(C(CC(C)C)N(C)C)=O)C(C)C2)=O)onc2ccccc12 c1(C(N2CC(CNC(=O)CCc3cccs3)OCC2)=O)c[nH]nc1[N+](=O)[O-] c1(C(C)C)cnc(C(c2nnnn2CC2CC2)NC2CC(n3ccnc3)C2)o1 c1(NCC23CC(N(C(CCC=C)=O)C(C)=O)(C2)C3)c(F)cc(C#N)cc1Br C(CC(N)=O)(C(=O)N(C)CC12CCC(CC1)CC2)NC(C(n1ccc(C)n1)C)=O Cc1ccccc1Sc1ccco1.c12ccc(cc1)NC(=O)NCCS2 c1(C(=O)OC)ccc2c(C)nn(C3(C(F)(F)F)CCCC3)c2c1 CC(C)C(C(C)C)C(C(=O)NCCC1CC1)N(C)CC12CCCCC1C2 C1(OC)(CNC(=O)NC(C(F)(F)C(F)(F)F)c2ccccc2)CCCS(=O)(=O)C1 c1(C(=O)NCCCCNC(COCC(=C)C)=O)ccc(C#CC2CC2)cc1 C1(CNC(c2c(C)snc2)=O)CN(C(c2cc(Cl)ncc2N)=O)C2COCC2O1 N1(C(c2cc(CCOC)on2)=O)CC2CC(NC(c3cocc3C)=O)C(C2)C1 C(=O)(C(C)(O)C(C)(C)C)N(CCC(C)NC(c1c(C)c(Cl)cnc1)=O)C c1(C(N(C2CCN(C(c3cnccc3Cl)=O)CC2)CC#C)=O)c(C)cccc1O CC1(CNC(=O)C2=COCCO2)CN(C(=O)CN2CCC(O)CC2)CCO1 N#Cc1ccc(OCC(N2CC(NC(=O)CN3CC4CCC3C4)C3CC23)=O)cc1 c1(CC(=O)NCC(C)(C)NC(C2(O)CCSC2)=O)coc(C2CC2)n1 C1(NC(C(CSC)O)=O)CC2COCC(C1)N2C(C1C2(CC2)C12CC2)=O c1(OC)cc(C(=O)NCCCN(C(=O)CC2CCC(C)O2)CCO)ccc1C c1(COC2C=CCOC2)ocnc1C(=O)NC(=O)NOC1CCOC1 C1(C(=O)NCC(CNC(c2cccc(CSCC)c2)=O)O)CCc2nnnn2C1 c1(NC(C(N(C(C(C)=CC(C)(C)C)=O)C)C2CC2)=O)ccc(Cl)nc1 CN1CCC(CC(=O)NC2(CNC(=O)C=Cc3cn[nH]c3)CCCC2)CC1 C1(CNC(C2C(C(C)C)(OC)C2)=O)CC(OC)CN1C(=O)CN(C)C(C)=O N1(C(C(C)C2CCCC2)=O)CC2CC1CCN2C(C1CCC1)=O C1(C(N)=O)CCC(C(=O)N(C2CC(NC(=O)COC3CC=CC3)C2)CCO)C1 c1(C(N2CC(NC(c3ncc(C)nc3)=O)C(F)C2)=O)c(Cl)ccc(Cl)c1F N1(C(C(C)=C2CCC2)=O)CCC(C(=O)NOC2CCOC2)CC1 C1(C(N2CC(O)(CNC(c3c(C)n(CCO)cc3)=O)C2)=O)CC2(CC2)CN1C C1(CNC(C2(C)CCN(C(C3CC4(CC4)CO3)=O)C2)=O)CC(C2CC2)=NO1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2CC(C1)N2C(=O)Cn1ccnn1 C1(NC(c2n[nH]c(CC)c2C)=O)CC2CC1N(C(c1cnn(C)c1C1CC1)=O)C2 C1(C(N(CCCN(C(C2(CC#C)CCCCC2)=O)C)C)=O)CCCC(=O)CC1 c1(C(=O)NC23CC(CNC(COCCOC)=O)(OC2)C3)cc(F)ccc1O c1(C(N2C(CNC(C3CC4CC3CC4O)=O)CCCC2)=O)cnc2ccnn2c1 C(C1CCCCC1)=CC(=O)NCC12CC1CN(C(C1(CO)CC(F)(F)C1)=O)C2 N1(C(c2c(CC)noc2C)=O)CCC2(CCC(NC(=O)C=Cc3cnc[nH]3)C2)C1 N1(C(c2nc(C)n(C)c2)=O)CC2CCC(C(=O)NCC3CCCC(C)(C)C3)(C2)C1 Cc1cc(C(=O)NCCC(C)N2CCCC2)c2cccc(C)c2n1 C(=O)(C(C)(C)CN(C(=O)Cc1cc(C)on1)C)NCC(C(C)C)OC C(=O)(C#Cc1ccccc1)NC1CN(C(c2ccc(C#C)cc2Cl)=O)CC1F C(=O)(C1CCc2snnc21)NC1CC2CN(C(CN(CCCCCC)C)=O)CC21 C(=O)(C(C(C)C)N(C)C)NC(C(=O)N1CC(F)(C(=O)OC)C1)Cn1cccc1 C1(NC(CC=CCC)=O)CCOCC1NC(c1cnn(C(C)C)c1Cl)=O c1(C(N2CC(NC(c3c(C)onc3Br)=O)C2)=O)ccc2[nH]ccc2c1F C(C)(C)(CCCC(=O)NC1(C)CCC(=O)NC1=O)NC(C=CCOC)=O C1(N(C)C)(NC(C2C=CCCC2)=O)CCOC1 S(=O)(=O)(c1cccnc1)CC(=O)NC(CN(C(CC(C)(F)F)=O)CC(C)(C)C)CO N1(C(C(C)NS(C)(=O)=O)=O)CC2(C1)C(NC(=O)NC(C)(C)C)C2(F)F c12c(sc3c1CCC(C)C3)NC2=O.C1(C)(CCC)CC(NC(=O)NC2CC2)C1 Cc1noc(C)c1-n1nc(-c2nc[nH]n2)nc1Cn1nnc(-c2ccco2)n1 C1(C(=O)NC2(CNC(CC3(C)CCCO3)=O)CC2)CCc2nccn2CC1 Nc1ccc(C(=O)NC2(CCNC(C3CCCOCC3)=O)CC2)c2cnccc12 C1(CC(N2CC(O)(CN(C(COCCCC)=O)C)C2)=O)SC2=NCCN2C1=O C1(NC(C=CCN(C(C(CC)OC)=O)C)=O)COC2(CCC2)C1 C#CC1C(C(=O)NC2CN(C(c3c[nH]nc3C3CCCC3)=O)CC2SC)C1(C)C c1(C(=O)NC2CC(C)(NC(CC3C(C)(C)C(O)C3)=O)C2)c[nH]c2cccc(F)c12 C1(CC)(CNC(=O)CCF)CCN(C(c2cn(C)nc2C2CCCC2)=O)CC1 c1(C(N2CC(CN(C(CC(CC)C)=O)C)C2)=O)cnc(Cl)cc1Cl C=C(CNC(=O)CCN1CCC(F)C1)CCNC(c1c[nH]cc1C(C)(C)C)=O c1(CCC)nc(C(=O)NCC(C)(C)CN(C(=O)Cc2nocc2C(C)C)C)co1 c1(C(C)NC(=O)CCC23CCC(CC2)C3)ccc(SC(F)(F)F)cc1 C1(NC(C(C)(C)Cc2cnn[nH]2)=O)CC2C(C1)C2(F)F.N12CCN(CC1)CC2=O CC1CN(Cc2c(C(=O)NCc3ccccn3)cc(F)cc2)CC(C)O1 C#CC1(CNC2CC(CC#N)C2)CCC1 C(=O)(C1=Cc2ccccc2C1)N1C(C)CC(Nc2ccc(OC)cc2[N+](=O)[O-])C1 c1(CN2CCC(NC(c3ccc(F)cc3I)=O)C(O)C2)csc2ccc(Cl)cc12 C1(C(=O)NC(CC#C)C(=O)OC)CN(C(=O)C(O)COC)C2(CCC2)C1 c1(C(N2CCC(F)(CNC(Cc3cnc(C)[nH]3)=O)C2)=O)c(S(N)(=O)=O)cnn1C c1(OC)ccc2ncccc2c1C(N1CC(CO)(NC(=O)CC(C)(C)SC)C1)=O C(=O)(C(O)CN(C)C)NC(C)C(C)NC(=O)CCOC1COC1 CCCCC(C)C(=O)N1CCC(CNC(=O)C(=O)NN(CCCC)CCCC)CC1 C1(NC(=O)CC2CCC(=O)N2)CCCCC1N(C(=O)C=C(Cl)Cl)CCO c1(C(N(CCCCC)CCO)=O)cc(C)n(C2CCCOC2)c1C C(=O)(C(F)C(=O)N1CC(NC(c2cc(Br)co2)=O)C(F)C1)OCC Cc1nnc2n1CCN(C(=O)C#CCNC(C1CC3CCC1CC3)=O)C2 N1(CCN(CCC)CC)CCC2(CCCN(C)C2)C1 N1(C(CC(COC)NC(=O)C2=NNC(=O)C2)=O)CC2(CC2)CC1C c1(C(=O)OC)nn(C)c2c1C(Nc1cc(Cl)c(Br)c(Cl)c1)CC2 Cc1cc(C(=O)Nc2ccc(-c3ccc(O)c(C#N)c3)cc2)c2nccn2c1 C1(NC(C=CCOC)=O)CN(C(c2n[nH]c(O)n2)=O)C2(CCC2)C1 CCC(C)C(C(=O)NCC(C)C(=O)OC)N(C(=O)Cc1nocc1C)C c1(OCC(N2CC3CC2CN3C(=O)C2=CSCCO2)=O)ccc2c(c1)CCC2 n1(CC=O)cnnc1O.CC(C)(C)SC1(CN(C(=O)CC2CC2C(F)(F)F)CC)CC1 C(C(CC(C)C)C(=O)NCCCC1C=NNC1=O)NC(CCCC(C)C)=O C=CCCC(O)CNC(=O)CCC1(NC(C2C3CCCC23)=O)CCC1 C1(NC(=O)Cc2ccoc2)CC(O)CN(C(c2cnn(CCO)c2)=O)C1 C=C1CC2(C1)CC(C(N1CCCC(NC(=O)C(c3cccc(O)c3)C)C1)=O)C2 c1(NCC2(F)CCN(C(C)C)CC2)ccc(CNS(=O)(=O)CCCl)c(Cl)n1 c1(C(N2C(CNC(CCSCCOC)=O)CCC2)=O)sc(N2CCCC2)nc1C C1(C(=O)NCCC(C)(C)N(C)C)CC(NC(c2ccc(=N)[nH]c2)=O)CCO1 c1(N(C)C)ccnc(C(=O)NC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)c1 c1(C(N(CC(CN(C)C(c2nc(Cl)cs2)=O)O)C)=O)cccc2c1OCCC2 C(C(C)(C)CCNC(C1CC(n2cnnc2)C1)=O)NC(c1c(C)[nH]cc1)=O c1(CNC(=O)C=CC2CC2)ccc2c(c1)CN(C(=O)C#CC1CCCOC1)C2 CC1CN(C(C2(c3cccs3)CC2)=O)CCCN1C(C1CC1N(C)C)=O C1(SCC(=O)NCCCNC(=O)CCc2ccc[nH]2)CCOC1=O C1(C(=O)NCC2(O)CCN(C(C34CCC(C3)C4)=O)C2)(CC)CCNC1=O Cc1nc(CC(=O)NCC(C)(C2CC2)NC(=O)CC(C)(F)F)c(Br)s1 C1(NC(=O)Cc2nnc(O)s2)CCN(C(=O)CNC(C2CCCC2)=O)CCC1(F)F c1(CCCC)nc(-c2ccoc2O)n(C2CCC(C)C2)n1 C1(NC(=O)COCC2CCCC2)CC2(CCN(C(c3ccc(Cl)nn3)=O)CC2)C1 C12(C(=O)NCC(CNC(c3cc(N)cc(F)c3)=O)CO)C3CC(CC13)C2(F)F C=CCC(C)C(=O)NCc1ncc(C(=O)N(C(C)C(C)C)C2CC2)cn1 c1(OC)ccc(Br)cc1-n1cc(-c2ccc(C#N)o2)nn1 CC1CN(C(c2cnc(O)s2)=O)CCCN1C(c1cn(CCO)nn1)=O N#Cc1ccc(NC(c2csc(C(=O)Nc3ccccc3O)n2)=O)c(I)c1 c1(CCC)ccccc1CNCC1CCN(CC#N)C1C c1(C(=O)NC(C(C)NC(C(C)NC(=O)NC)=O)(C)C)ccc(C(N)=O)c(Cl)c1 CC1c2c[nH]nc2CCC1C(N1CCOC(CN(C(=O)CSC(F)(F)F)C)C1)=O CCC(CC(F)F)C(=O)N1CCCC(N(C)C(c2coc(C(C)(C)C)n2)=O)C1 Cc1noc(C)c1C(N1CC(CNC(c2ccoc2C2CC2)=O)C(O)C1)=O N1(C(C(C(=O)OCC)F)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)CC)CCO2 N1(C(c2c(F)ccc(OC)c2)=O)CC(C)OC2(CCN(C(=O)C(C)(C)OC)C2)C1 c1(SCCCC)cccc(C(N2CC3CC3(NC(C3CCN(C)CC3)=O)C2)=O)c1 C1(NC(Cc2c(C)cccc2)=O)CC=C(C(=O)N2CCC(OC(C)C)C2)C1 C#CCC(C(=O)NCc1ccn(C2CC2)n1)NC(C1CCC1)=O C12(NC(CCC=C=C)=O)CCCCC1N(C(=O)Cc1cnccn1)CC2 C1(CC#C)(C(N2CC(C)(CC)C2)=O)CCN(C(C2OC3CCC2C3)=O)C1 c1(OC)cc(C=CC(=O)N(C(C)CNC(c2cccnc2C)=O)C)sn1 Cc1ccc(F)c(C(C(=O)NCc2ccccc2)N(CC(F)Cl)C)n1 c1(C(N2CCC3C(CCN3Cc3cc(Cl)ccn3)C2)=O)cc(I)ccc1[N+](=O)[O-] N1(C(c2ccc(C3CC3)c(Cl)c2)=O)CC2CCCOC2C1 N1(C(c2cnc(-c3ccccc3)cn2)=O)CC2COC(C1)C2O N1(C(CCCc2onc(C)n2)=O)CC2CC(NC(C34CCCC(C3)OC4)=O)C1C2 Cc1cc(F)c(C(=O)NC2CC3CN(C(=O)CN4CC=CC4)CC3C2)cc1Br c1(NC(C(n2ccc3ccccc3c2=O)C)=O)cc(Br)cc([N+](=O)[O-])c1 c1(OC)nc(C)ccc1C(N1CCC(CO)(NC(C2C(C)(C)C2(F)F)=O)CC1)=O C1(c2onc(C(C)(C)C)n2)CCN(C(=O)CC(N)CO)CC1 c1(OCC)ccc(COC(=O)C(CC(C)=O)NC(=O)CC(F)(F)F)cc1C C1(F)(CNC(C(COCC=C)C(C)C)=O)CCCN(C(C2C3CCCC23)=O)CC1 C#CCCCCCCC(=O)N1CCC2(CCC2)C(NC(=O)C(C)C(C)O)C1 CCCC(CC1CCCC1)C(=O)N1CC(CNC(=O)C(C)N(C)CC)(OC)C1 c12cnc(nc1)CNC2=O.c1(C(C)C(=O)NC(c2nncs2)C)ccccc1 C1(N(CC(C)C)CCO)CCN(C(=O)C(C)C2CCOC2)CC1 C(=O)(CC(C)(C(F)F)N(C)C)NC(c1ccccc1)CNC(c1ccc(C)n1C)=O CC(C)(C)CC(F)C(=O)N1CCCC(CC(=O)NCCC(O)CCO)CC1 C(=O)(C#CC1CCCCC1)N1CCCC(NC(C(COC)(C)C)=O)C(F)C1 c1(C(=O)NCC(C2CC2)NC(=O)C(O)C2CC2)n[nH]c2c1COCC2 c1(C(N2CC(OCCNC(C(CC)OCC)=O)C2)=O)ccc2[nH]cc(C#N)c2c1 c1(C(N2CC(CN(C)CC)C2)=O)ccncc1.C(C(F)(F)F)NCC(=O)N CCC(CC)CC(=O)NC12CCN(C(=O)Cn3nc(C)cc3C)CC1C2 C(=O)(C1COc2ccccc21)NCC(CNC(=O)C(C)(C)CS(C)(=O)=O)OC C(C(=O)C(C)(C)C)N(C(C(C)(C)OCNC(C)=O)=O)C C(CC(C(C)(C)C)N(C(=O)OC(C)(C)C)C)OC.C1=[SH]C1(C)C.C(=O)O c1(CN2CC3C(C(=O)Nc4cnc(OC)nc4)(C3)C2)ccnc(F)c1Cl CC(CCCN=c1ccc(-c2ccccc2)n[nH]1)NC(c1cc(Cl)on1)=O c1(C(N2CCCCC(NC(CC(CC)O)=O)C2)=O)cnc2ccccc2c1C N1(C(C(C)OCC2CC2)=O)CCOCCC1C(=O)NCC=CC1CC1 c1(CCC)cc(C(=O)NC(CNC(=O)CC2CCCCC2)CC)no1 CC1=C(C(=O)N2CCN(C)C(C(=O)NC(C)(C)C(=O)N(C)C)C2)CCO1 c1(C2(C(N3C(C)CC(CNC(C(OC)OC)=O)C3)=O)CCC2)ccc(Cl)c(F)c1 C1(CNC(c2nc(CSC)sc2)=O)CC2CCC1N2C(=O)CSc1cccs1 c1(C=O)cnc(CC)s1.C1C(C)(OCC)CNN1CCOCCOCC.C1CC1 N1(C(CCc2cc(C)no2)=O)CC2CC2(NC(=O)CCCc2ccccc2)C1 C1(NC(CC2(C)CCCCC2)=O)C2CC3C1C3C2C(=O)NCC#CCCO c1(C(C(=O)NCC(CC)(C)NC(c2csnn2)=O)OC)ccc(Br)cc1 c1(C(=O)NCC2(CNC(C(CC(C)C)N(C)C)=O)CC2)coc2cc(F)ccc12 N1(C(C(C)(C)OC)=O)CCC(C)(CC(=O)N(C)CC2CCC(C)CC2)C1 n1(CC(=O)NC(C2CN(C(=O)COc3ccc(Cl)nc3)C2)C)cccnc1=O C1(O)(COCC(=O)N(C2CCCOC2)CCOCC)CCN(C2CC2)C1.CC C1(C(=O)NCCC2CC(NC(=O)CCOC3CCOCC3)C2)CC2(C1)CC2(F)F c1(C(N2CC(C)(C)OCC2CCO)=O)ccc2c(c1)CCOC2 c1(NC(=O)NC(CCC=C)c2ccccc2)c(Cc2ccccc2)noc1C Cc1nsc(C)c1C(N1CC(CCCCNC(C2CCCCN2C)=O)C1)=O N1(C(CC(=O)OCC)=O)CC(NC(=O)C(C)N(C)C)C(C)C1 c1(N2CC(C(C)NC(=O)CCC[N+](=O)[O-])C2)cc(C(F)(F)F)ncc1[N+](=O)[O-] C#CC12C3C4C1C1C2C3C41C(=O)NC1CC(F)(CNC(=O)CC(=O)N(C)C)C1 C(C)(C(CC(=O)N1CCCCC1C)NC(=O)CCC(=O)C1CC1)OC C1(NC(C2C3(CCN(C(c4ccc(OC)s4)=O)C3)C2)=O)Cc2ccccc2O1 C1(C(N(C2CC3(CCC3)C2)C)=O)CC2CCCC2N1C(c1cccc[n+]1[O-])=O n1(CC)cccc1C(=O)N(CCNC(C1CCCN1C1CCCCC1)=O)C1CC1 C1(C(=O)NCCC2CC(F)(F)C2)CC(F)CN1C(=O)C(F)CC1CCOC1 C1(O)(CNC(CCC(C)OCC)=O)CCCN(C(=O)COCCSC)C1 C1(CC)CN(C(=O)CC2CCCOC2)CC1C(=O)NC(CC1CC1)C1CC1 c1(C(=O)NCC2C(C)CCN2C(=O)C2CC2)cc2n(n1)CCO2 c1(C(=O)NC23CC(C(=O)Nc4ncc(Cl)nc4Cl)(C2)C3)ccc2ocnc2c1 CC1CCC(=CC(=O)NC2CN(C(C3CCN(CC(C)C)C3)=O)CC2F)CC1 N1(C(C2C(C)OCC2)=O)CCC(CO)CC1.c1(CN)cnn(C(C)(C)OC)c1Cl N1(C(CC(CCC)O)=O)CCCC2(CCN(C(C3(C)CC3C)=O)CC2)C1 N1(C(CC(=C)C)=O)CC2C(CNC(c3ccc(-c4cccn4C)cc3)=O)C2C1 c1(OC)c([N+](=O)[O-])ccc(CSC2N(C(=O)Cn3ccnc3)CC2(C)C)c1O CC(C)(O)C(F)C(=O)NCC1CCN(C(C23CC(c4ccccc4)(CO2)C3)=O)C1 c1(CC(=O)N(CC(C)CNC(=O)CC2CCCO2)C)cc(F)cc(Cl)c1 c1(OC)ccc(F)c(C(c2nnnn2CCCF)Nc2ccsc2)c1F C1(C(N(CC(O)CNC(=O)Cc2ccccc2Br)C)=O)Cc2nncn2C1 C1(C(=O)NCCCCC(=O)NCCN2CCOCC2)Cc2ccccc2C1 c1(CNC(N2C(C)(COC)CC2)=O)cccc(OC)c1 c1(CCC)[nH]ccc1C(=O)NCC(C(=O)NCCN1CC=CC1)N(C)C c1(C(N(C2CCN(C(=O)C=C(C)C3CC3)C2)CCC)=O)cc(OC(F)F)ns1 N1(C(CCC(CC)OC)=O)CCOC2CCN(C(c3ccc(F)s3)=O)CC12 c12ccccc1CC(=O)NCC2.C(CC(C)NC(C1(SC)CC1)=O)SCC Cc1cc(CN2CCOC(CC(=O)NC3CNC(=O)C3)C2)ccn1 N12CCN(CC1=O)Cc1ccc(o1)C(=O)C(=O)C2.n1(C(C)C)cc(CN)nn1 C(CN=C(NCC(CO)C1CC1)N1CC(O)C(C)(C)C1)OCCOC C1(C(=O)NCC23OCC(NC(C(C)OC)=O)(C2)C3)CC2CCCC2C1 CC1(NC(C2CC(C3CC3)=NO2)=O)CCN(C(c2cn(CC3CC3)nn2)=O)CC1 C(=O)(C(C(C)(C)C)n1ccnn1)NCC(C)CN(C)C(C1CC(=O)NC(C)C1)=O C1(CS(C)(=O)=O)CN(C(=O)Cc2ccco2)CCN1C(C1CCCO1)=O N1(C(CCNC(C)=O)=O)CC2CC(C(N3CCC(C)(CO)C3)=O)(C2)C1 c1(C(=O)NCC2(CNC(=O)CCCc3cnn[nH]3)CC2)ccccc1OCCF Cc1cccnc1CCC(=O)NCC(C)NC(c1ccccc1CC#N)=O N1(C(CC(CNC(C2N(C(C)C)CCC2)=O)(C)C)=O)CCN(C)CC(O)C1 c1(N(C(=O)NCCNS(C)(=O)=O)C)c(N)cccc1Br C(CC(=O)NCC1CCN(C(c2c[nH]nc2C2CC2)=O)C1)(C(C)C)OCC CCCCC(C)C(=O)N(CCCC(=O)NCCC(F)=C(F)F)C(C)C CC(C)CC(CNC(=O)COCCNC(C1(CCOCF)CC1)=O)CO C(=O)(C1=CC2CCCC12)N1CC2C(NC(c3cc(OC)no3)=O)(C2)C1 n1(CCNC(C(C2CCN(C(C=CC(CC)C)=O)C2)C)=O)cnccc1=O CC(N=c1cc[nH]cc1S(=O)(=O)NCC1(F)CC(O)C1)c1ccsc1 C1(C(=O)NCCC2N(C(Cn3c(C)nnn3)=O)CCSC2)CCCCC12CCC2 C1(CNC(CN(CCC)C)=O)CC2COCC2N1C(c1cc(CC)ccc1O)=O N#Cc1cc(NCC2(c3ccccc3)CCOC2)cc(Br)c1 N1(C(CC2CC(OC(C)(C)C)C2(C)C)=O)CCCC2(C1)CN(S(=O)(=O)C1CC1)C2 C1(C(=O)NCC2C3CN(C(=O)C4CC4)CC23)CC(c2cccc(Cl)c2F)=NO1 N1(C(COC2CN(C(C3C(C)OCC3)=O)C2)=O)CCOC(C(C)(C)C)C1 c1(C(=O)OC)ccc(CNC(C2CC(CNC(C3COC(CO)C3)=O)C2)=O)cc1 c1(C(=O)NCCC(=O)OC(C)C)cnc(CNC(C2(C)CCCC2O)=O)nc1 C(c1cc(F)cc(F)c1)=CC(N1CCC(NC(C(CC)NC(N)=O)=O)C1(C)C)=O Cc1cc(C(=O)NC2(C)CCN(C(=O)CCCC3CC3)C2)c2cccc(C)c2n1 CC1(NC(=O)CCc2ccc[nH]2)CN(C(=O)CSCC(F)F)C1 C#CCC(C)C(=O)N1CCCC(CN(C(=O)CN(C)C(c2ccsc2)=O)C)C1 N1(CC(N2C(C(=O)NC3CCN(C)C3=O)CC=CC2)=O)C(=O)CCCC1=O c1(C(=O)NC2CN(C(c3c(C)c(Cl)ccn3)=O)CC2C)ccc2c(n1)CCCN2 C1(CC(N2C(CNC(c3n(C)cc(Cl)c3)=O)CCC2)=O)COCC(C)(C)O1 c1(C(=O)NC(C2CN(C(=O)CCc3cn[nH]c3)C2)C)cc(C(F)(F)F)cs1 N1(C(CN(C(C(C)C)=O)C)=O)CCOCC(NC(=O)CCc2cccn2C)C1 C1(NC(C(c2ccc(C#N)s2)(C)C2CC2)=O)CCCCC1n1cccn1 C1(C(=O)NCCOCCC)CC2CCN(N(C3CCCC3)C)CC12 c1(C(N2CC3C(NC(CCC(CC)CC)=O)(C3)C2)=O)ccc(F)c(S(N)(=O)=O)c1 C1(C(N(CCNC(C(CC)n2nccc2C)=O)CCOC)=O)COC(C)(C)CO1 O=C1CN(C(=O)CCS(N)(=O)=O)C2CCN(C(C3Cc4nccn4C3)=O)CC2N1 C#CCC(C)C(=O)N1CC2(NC(c3sc(OC)nc3Cl)=O)CC1C2 C(=O)(CCC(=O)N1CC1)NCC1N(C(C2N(C(C)=O)CSC2)=O)CCC1 N1(C(C(C)CN(C)C)=O)CCCC1(C)CNC(C1(n2ccnn2)CC1)=O N1(C(C(C=CC)O)=O)CCCC1(C)CNC(=O)CSCCN(C)C c1(C(=O)NC(C)CCNC(=O)C(C)CO)cc(Cl)cc(Br)c1 Cn1cc(S(N)(=O)=O)c(NC2CCCCC23CCC3)n1 c1(CCC(=O)N(CCC(=O)NCC(c2cccnc2)C)CCCO)ccn(C)n1 c1(C(=O)NC2CN(C(CCC(=C)Cl)=O)CC2CO)ccc(F)cc1C#N C1(C(C)C)(C(=O)NC(C)CC2CN(C(=O)CCNC(=O)C=CCl)C2)CCCO1 c1(OC)ccc(C(=O)NCC(F)CNC(=O)CCc2ncc[nH]2)cc1C1CC1 C(=O)(C1Cc2c(Cl)cccc21)NC(CNC(c1ccc(CC#N)cc1)=O)C1CC1 C#Cc1cncc(C(N2CCN(C(=O)CC3CCCC(C)(C)C3)C(C)C2)=O)c1 N1(C(C(C)OC(c2c(C)onc2)=O)=O)CCC(C)N(C(=O)OC(C)(C)C)CC1 N1(C(c2ccc(N)cn2)=O)C2CCC(C(=O)NC3CC4(CCC4)C3O)C1CC2 c1(C(=O)NCC(C2CCC2)NC(=O)CCC2CCC2)ccn(C2CCCC2)n1 c1(C(=O)NC(CCCNC(CSC(C)C)=O)C)ccc(C(F)F)nc1O N1(C(CCc2ccc(C)o2)=O)CCC2CN(C(=O)CSc3ccccn3)CCC12 C1(C(=O)NCc2ccc(OC)c(Br)c2)CCc2nc(C)nn2C1 CCC(CCCC(=O)NCc1ccn(C(C)C)n1)NC(=O)Cc1ncccc1F C1(C(N(CCC(C)(C)NC(c2cncs2)=O)C)=O)CC2CC1C1CC21 C1(=CC(N2CC(C)N(C(=O)CS(C)(=O)=O)CC2)=O)CCCCCC1(F)F N1(C(C2(CC)CCOC2)=O)CCCC(F)(CNC(=O)C(C(C)C)N(C)C)C1 c1(C(N2CC(C)C(NC(C3CC(C)(C)C3)=O)C2)=O)ccc([N+](=O)[O-])cc1N c1(C(C(=O)N(CC(C)NC(c2cncnc2)=O)C)C)c(F)cccc1F C1(NC(Cc2c(OC)nccc2)=O)CCC2(CC1)CN(C(C1CC(C)=NO1)=O)C2 C1(NC(C=C(CC)CC)=O)CC(O)CN(C(=O)Cc2cnccc2C)C1 N1(C(C(C)Cn2cccn2)=O)CC(C2(NC(C3CCCC(O)C3)=O)CC2)C1 c1(C(=O)NC(CNC(c2c(C(C)C)ocn2)=O)C)nn(C)c(Cl)c1Cl C1(CNC(c2cccs2)=O)CN(C(C2CC3(CC3)CO2)=O)CC12CCOCC2 C(C)(C(C)CC)(c1ccccc1)N(C(C(C)SC)=O)C.n12cc(nn1)CCCC2 C1(CCN=C(NC2C(C)C2)NCC(C)(O)CN2CCOCC2)CC2CCC(C1)N2C CCC(C(=O)NCC1CC(NC(c2cnn(-c3cccc(F)c3)c2)=O)C1)C(C)O CCC(CC(F)F)C(=O)N1CC2(CCC2)CC1CNC(c1cnc(S)nc1)=O C1(NC(CSc2cccc(C)c2)=O)CC2CCC1N2C(=O)Cc1cc(Cl)n(C)n1 C1(C(N(CCCC(=O)N(C)C)C)=O)CCC2CCC1N2C(C12COCC1C2)=O c1(CCC)[nH]ccc1C(=O)NCCNC(=O)C(C1CC1)OCc1scnc1C.OC c1(C(=O)NCCC2CCCN(C(C(C3CC3)OCC)=O)C2)cncc(N)c1C c1(C(N2CCC(CNC(CC3C(C)(C)CCC3)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] n1(CC(N2C(CCNC(C(F)=CC)=O)CCCC2)=O)cc(Br)c(O)nc1=O C12(NC(C(C)(C)OC)=O)CCC(CC1n1cc(C3CC3)nn1)C2.N1C(=O)CCC1=O C1(CCNC(C2CC23CCOC3)=O)CCN(C(C2CC3(CC3)CO2)=O)CC1 C(c1ccc(Br)cc1F)=CC(N1CC(F)(CSC)C1)=O.c12n[nH]c(c1C#N)NC2=O Cc1cccn2c(=O)cc(CNCC(O)Cc3ccc(F)cc3F)nc12 C1(C)(CN(C(=O)CC2CCCC2)C)CCCC1NC(=O)CC1CCCO1 C(=O)(C1=NOC2COCC12)NCc1ccc(C(N(C23CC(C2)C3)C)=O)cc1 Cc1cc(CC(N2CC(O)(C(C)NC(=O)COc3ccccc3)C2)=O)ccc1O N1(C(CCC(=O)N(C)C)=O)CCC(NC(=O)CSC(F)(F)F)C(O)C1 c1(C(=O)NC(CNC(c2c(C)cccc2)=O)C2CC2)ccnc(C)c1N C1(C(=O)NC2(C)CN(C(C3OCCOC3(C)C)=O)C2)CC2C=CC1CC2 c1(N2CC(NC(c3cnn(C(C)C)n3)=O)C(C)(C)C2)ncc(Br)cc1[N+](=O)[O-] CCC(O)C(C)C(=O)N1CC(CNC(=O)C(F)(F)CC2CC2)C(C)C1 C1(C)(C(N2CC(CCNC(C#CC3(CC)CC3)=O)OCC2)=O)CC(C(C)C)=NO1 C(=O)(C(F)C(=O)N1CCCCC1CCNC(c1cnc(S)n1C)=O)OCC CC(C)(C(=O)NC1CC(COC(c2ccc(Cl)c(C(CCCCN)ON)c2)=O)C1)C(N)=O C1(C(=O)NC2CCC(NC(COC3(C)CCOC3)=O)C2)NC(=O)CC1(C)C N1(C(C#CCNC(c2cc(OC)no2)=O)=O)CCCC(F)C1 N1(Cc2nnc(C)s2)CCC(n2cc(C(=O)NCc3cccc(F)c3)nn2)CC1 N1(C(C(C)OC2CCCC2)=O)CC(NC(c2csc(Cl)c2Cl)=O)C(C)(C)C1 CCS(=O)c1ccc(-c2ccc(C(=O)Nc3cc(Cl)c4cn[nH]c4c3)nc2)cc1 C1(N(CC(C)(C)O)C(c2c(C(C)C)onc2)=O)CCNCC(C)(C)C1 S(=O)(=O)(c1ccc2[nH]c(=NC3COC(C)(C)C3)ccc2c1)NCCCC(C)O c1(C(=O)NCCN(C(C2CC2C2CCCO2)=O)C2CC2)c(Cl)ccc(Cl)c1O N1(C(=O)NC(C(=O)NC)Cc2ccccc2)CCCCCC1C(C)(C)C c1(NC(=O)CCSCN(C(CC)C(=O)NC2CCC3(CC3)C2)C)oc(C)nc1C#N C1(CNC(COCCCN=[N+]=[N-])=O)CC(C(=O)NCCS(C)(=O)=O)=NO1 N1(C(CN(C(c2cc(CC)[nH]n2)=O)C)=O)CCN(C(c2cc(C)[nH]c2C)=O)CC1 Cc1cccc(Br)c1C(C(=O)NCCC1OCCC1(C)C)NC(=O)C(F)F N1(C(CC(C=C)C)=O)CCN(C)CC1CNC(=O)CNC(=O)C(CC)CC C1(NC(c2nc(C)[nH]c2C(F)(F)F)=O)CN(C(c2cncnc2C)=O)CC12CC2 C1(CC(=O)N(CCNC(c2nncs2)=O)CC)CC2COCC12 N1(C(CC2N(C(C3CC4CC(=O)C3O4)=O)CC(F)C2)=O)CCC2(CC1)CC(O)C2 N1(C(c2cccc[n+]2[O-])=O)CCCC2(CCN(C(=O)C(F)(F)CF)C2)C1 C(C(C(F)(F)F)N1CCNCC1)NC(C(=O)NCCCSCC)=O C(=O)(C(C)(C)C(=O)NC1CC1C(=O)NCC(C)OC(F)F)OC N1(C(C2CC(CNC(c3cccc(C)c3O)=O)OC2)=O)CCOC(C)(C)C1C Cc1cc(C)c(NC(C2CCCCC2NC(c2ccc(F)c(Br)c2)=O)=O)cc1Br c1(CN2CCC(C)(CC)C2)cnn2cccc(-c3cc(C)cnc3F)c12 C1(NC(C(COCC)NC(C2CCC(CO)C2)=O)=O)CC(CO)C12CCC2 C12(C(N(CCCCNC(C(CC(C)C)N(C)C)=O)C)=O)CC1Cc1c[nH]nc12 Cc1nc2cc(NC(C3CCC(NC(c4n[nH]c(C)c4C)=O)CC3)=O)cnc2[nH]1 CCS(=O)(=O)CC(=O)NCCCCC1CCN(C(c2cccc(C)c2Cl)=O)CC1 C1(C(N2C(CC)CCC(C)C2)=O)CN(CC)CCC1O c1(C(=O)OC)ccc(C2(C(N3CCC(N(C(=O)C=NOC)C)C3)=O)CC2)cc1 CC1=NN(C)C(=O)C1CC(=O)NCC1(CN(C)C(C2CCC(C)(C)OC2)=O)CC1 c1(C(C#C)Oc2cc[nH]n2)cc(F)cc(F)c1.N12CCN(CC1)CC2=O C1(NC(C2CCN(C(=O)NC)C2)=O)CCC(NC(C2COCCN2C)=O)CC1 c1(C)cc(C(N2CCCC(NC(c3ccc(SC)cc3)=O)C2)=O)sc1C.CO Cc1nc(=N)[nH]c(=NCC2(c3ccc(Cl)cc3)CC2)[nH]1 CCC(CC(=O)N1CCCC(O)(CNC(C2C(Cl)(Cl)C23CC3)=O)CC1)C(C)C c1(C(=O)NC(CCCNC(C2(CCC=C)CCCC2)=O)C)cccc(O)n1 C1(CCC)CN(C(=O)CC(C)OC)CC1NC(c1cc(C(CC)CC)no1)=O c1(CC)ccc(O)c(C(=O)NCC(C)(C2CC2)NC(C2CC=CCC2C)=O)c1 CC1C(C(=O)Nc2nnccc2C(F)(F)F)CCN1C CCC(C(=O)N1CCC(NC(=O)COc2cc(C)on2)C1)C(F)(F)F N1(C(C2(OCC)CC2)=O)CCC2(CCCN(C(C3COCCC3(F)F)=O)C2)C1 N1(C(CC(=O)OCC)=O)CCC(C2(NC(=O)CCCN(CC(F)(F)F)C)CC2)C1 C(=O)(C(O)CC(F)(F)F)N(C(C(=O)NCC1CCN(CC)CC1)C)C1CC1 c1(C(=O)NC(C)CNC(c2cc(C(=O)O)cc(Br)c2)=O)cc2cc(Cl)ccn2n1 C=CCC(CNC(=O)Cc1cncn1C)C(=O)NC1CC(CF)C1 C1(NC(c2scc3c2OCCO3)=O)COC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 N1(C(C(C)c2cc[nH]n2)=O)CCCC2C1CCCN2C(=O)CC1CSCCO1 c1(N2CC(CNC(=O)NC)OCC2)ccc(S(=O)(=O)NCC(CO)OC)c(Br)c1 Cc1cc(CNC2CC(C(=O)NCCC(C)(C)C)C2)c(C)cc1Br N1(C(C(=O)NC(CC)(C)C)CC(C)C)C2CCC1c1ccccc12 C(C)(CNC(C1C2CC3C(C2)C13)=O)(CC(C)C)NC(c1c(C)n(CCO)cc1)=O CN1CC(C)(C(=O)NC(CO)C(=O)N2CCC2CF)CC1=O N12CCC(CC1)C2=O.CC(CC(=O)N1CCC(C(C)(C)C)C1)C1CC1 CN1CCC(O)(C2(C(=O)NCC(C3CC3)NC(=O)C=CC(=O)N(C)C)CC2)CC1 C1(CC(=O)N(CCF)CC)C2CN(C(=O)CC3COC(=O)C3)CC12 c1(C(C)N(C(=O)CC2CC=CC2)CC2CC2)ccc(Br)c(F)c1 c1(C(=O)NCC(C)CN(C)C(c2ccc(CO)c(F)c2)=O)n[nH]cc1[N+](=O)[O-] CC1CN2CCN1C(C(N1CC(N(C)C(c3nccn3C)=O)C1)=O)C2 C12(C(=O)NCCCCNC(CCC(C)(C)C#N)=O)CC3CC(C1)CC(C)(C3)C2 c1(CC)n[nH]c2cc(C3=CCCN(c4cc(C#N)ncn4)C3)ccc12.N1CCNCC1 Cc1ccc(C(=O)NC2CN(C(=O)CCSC3CCCC3)CC2C)c2c1CCC2 c1(OC)c(C(=O)Nc2cccc(C3CC3)c2)cccc1F C(=O)(CCS(N)(=O)=O)NC(CN(C(c1cc(CC)on1)=O)C)C N1(C(CC=CCC)=O)CC(C)(C)CCC1CNC(C1CCCC(F)C1)=O C(C(=O)N1CCC(NC(C2(C)CCC(OC)CC2)=O)C(F)C1)(C(C)(C)C)OC CC1CC(CNC(N2CCC(C(N3CCCC3)=O)C2)=O)=NO1 c1(C(N2CC3CC(CNC(C4CC4F)=O)C3C2)=O)nncc2ccccc12 C1(C(C)C)CCN(C(=O)CCC2CCN(C(=O)Cc3ncccn3)CC2)CC1 N1(C(C(=O)N(C)C)=O)CCCCC1c1n[nH]cc1C(=O)NCC1CCCCCC1 N1(C(C(C(C)OC)NC(=O)C=CC2CCCCC2)=O)CCCC(CO)CC1 C1(NC(Cc2nc(C)[nH]n2)=O)CN(C(C23CCC(CO)(CC2)C3)=O)CCC1(C)C c1(C(N2C(CNC(CN(C(c3c(C)occ3)=O)CC)=O)CC2)=O)cc(F)ccc1O N1(C(C(C=C)O)=O)CC(CNC(c2cc(O)ccc2C(C)C)=O)CC1(C)C Cn1c(C(=O)NCC2CC(NC(=O)Cc3ccc(F)c(CO)c3)C2)ccc1C#N n1(CC(N2CC(C(C)NC(C3CC3(C)Br)=O)OCC2)=O)ccc2ccccc12 c1(OC)ccc(C(=O)NC2CC(C)N(C(=O)CC3CSCCS3)C2)c(F)c1N N1(C(=O)C2=CC(O)CCC2)CCC2(C1)CN(C(C1(CC3CC3)CC1)=O)CCO2 c1(OC)cc(C(=O)NC(CNC(=O)C(O)C(C)(C)C)CO)c(F)cc1N N1(CC=CC(=O)NC(C)CCNC(C2CCC2C(F)(F)F)=O)CCOCC1 C12(C(=O)NC(CCCNC(c3ncc(OC)cn3)=O)C)CCCC1CCC2 C(C(C)(C(=O)N(CCC(=O)NCc1nc(C)sc1C)C)OC)OC c1(CSC)ccc(C(N2CC(CNC(c3nocc3C(C)(C)C)=O)C2)=O)cc1 C1(NC(c2c(C)nco2)=O)CCCN(C(C2CCCN(C(C)C)C2)=O)C1C CCCCC(CC)CC(=O)NCCC(C)(C)C(=O)NC1CC(OC)C1(C)C CC1CCOCCN1C(c1[nH]ccc1CNC(=O)CCCC1CCCC1)=O S(=O)(=O)(c1ccc(NCCCN2C(=O)CCC2=O)c(F)c1)NCC(CC(C)C)O c1(C(=O)NCC2CCC(NC(c3cn(CC)nc3C)=O)C2)ccc2[nH]ccc2n1 C1(NC(c2cccc(F)c2)=O)CC2CN(C(=O)CCn3cccnc3=O)CC2C1 C(=O)(C1=NOC(C)(C)C1)NCC1CC(NCc2n(C)nnn2)C(O)C1 C1(C(=O)Nc2ccc(CN(C)C)o2)CN(c2ncncc2I)CC(F)(F)C1 C1(COC)CN(C(C2CC(C(N)=O)C2)=O)CCN1C(=O)C(O)CN1CCCC1 C(CCCCC(=O)NC1CC(N(C(=O)C(C)C2CCCO2)C)C1)OC C1(NC(c2nnnn2-c2ncc[nH]2)=O)CCN(C(=O)C(=O)NCC(F)(F)F)CC1 C1(C)(C(=O)N)CC2C=CC1C2.C1(C(=O)NCc2cc(C)on2)CCC(CO)CC1 C1(N(C(CN(CCCN(C)C)CC)=O)C)CCCN(c2ccc(OC)cc2)C1=O C=CC1(C(=O)NC2(CCCF)CCC2)CCN(C(=O)Cc2n[nH]c(C)n2)CC1 c1(C(=O)OCC)cc(Br)cc(Br)c1NC(C1CCN1C(c1ccc(CC)o1)=O)=O C1(NC(Cc2c(C)scc2)=O)CCN(C(C2CCC(C)(C)O2)=O)CC1 C1(O)(CCNC(c2cccc(F)c2C(F)(F)F)=O)CCCN(C(C2CCC2)=O)C1 C#Cc1cccc(C(=O)N(CCCNC(c2ncc[nH]c2=O)=O)C(C)C)c1Cl S(=O)(=O)(c1ccc(NCC2(c3nnnn3C(C)C)CC2)c(Cl)c1)NCC(=CC)Cl N1(C(CNC(C)=O)=O)CCCOC(CNC(=O)Cn2ccccc2=O)C1 Cc1cc(NC(C2CCCC2CNC(=O)C(C2CCOCC2)C)=O)cs1 c1(C(=O)NCC2CCN2C(C2C3COCC23)=O)cccc2sncc12 N1(C(=O)NCc2csc3c(O)ccnc23)CCOc2ccc(C(F)(F)F)cc21 N1(C(C2C(NC(C(C)OCC(C)C)=O)CC2)=O)CCC2(CC1)CN(C)C2 c1(CC)cc(F)ccc1C(=O)NCCC(C)NC(=O)Cc1cc(Cl)cnc1C CC(CC(C)NC(C1CCC2CC12)=O)NC(=O)CCc1nccn1C C1(C(N2C(C)CCC(NC(=O)Cc3cnn(C)n3)C2)=O)Cc2ccncc2C1 c1(C(=O)NCC(N)=O)ccc(NC(=O)Nc2ccccc2)cc1 C(=O)(CC(O)CC(C)(C)C)N(CCC(c1cccs1)NC(C(COC)C)=O)C N#CC1(C(=O)NC23CC(C(N4CCC(O)(C(=O)NC)CC4)=O)(C2)C3)CC2CC2C1 n1(CC(=O)NCC2CN(C(CNS(N)(=O)=O)=O)CC2(F)CO)cc2ccccc2n1 c1(C(=O)NCC2CC(NC(C3COCC(C)O3)=O)C2)coc2c(Cl)cccc12 CC#CCC(C(=O)NCC1CN2CCC1C2)NC(=O)CCCOC(C)=O C(=O)(CC(C)C(F)(F)F)NC(C1(O)CCN(C(CCc2onc(C)n2)=O)C1)C N1(C(C(C(C)OC)N(C)C)=O)CCN(C)CC1C(=O)NCC(O)C(F)F C1(C(=O)NC(C)(C)CNC(c2cc3sccc3cn2)=O)CCCC12CCOCC2 c1(NC(C2(N(C(C=CCN(C)CC)=O)C)CC2)=O)cnc(O)c([N+](=O)[O-])c1 N1(C(=O)CSc2ncccn2)CC2CCN(S(=O)(=O)c3ccncc3)C2C1 c1(C(=O)NC(CC(C)NC(C2CCC(C(=O)OC)C2)=O)C)nccnc1OC C1(CCN(C(=O)C2=CCCO2)C)CCN(C(c2ccccn2)=O)CC1 c1(C(=O)NCC2CCN(C(c3c(OC)c[nH]n3)=O)CC2O)cccc2c1COC2 C(c1c[nH]c2ccccc12)=CC(=O)NC1C(C(N2CCCC(C)CC2)=O)C1 C1(NC(C=C(C)C)=O)CCCN(C(=O)C=CC2CCCO2)C1C c1(OC)cc(CC(=O)N(C2CN(C(=O)CC3CCOC3(C)C)C2)C)ccc1O Cc1cc(C(=O)NCCCN(C)C(C2CCCCC2O)=O)c(O)nc1C N1(C(c2cccc(Br)c2F)C(=O)NC(C(=O)OC)C)CCc2n[nH]cc2C1 C1(C(N(CC)Cc2ncc[nH]2)=O)CN(C(=O)Cn2c(O)nnc2O)CC1F c1(N)cc(Br)ccc1S(=O)(=O)Nc1cc(Br)cs1.C(C)(CN(CCO)C)OC C1(NC(C2(C)CCCC2)=O)CN(C(c2cc(Br)n[nH]2)=O)C2CCCCC12 C(=O)(CC(C(F)F)n1ccnc1)NCC1(NC(c2c(C)n(C)cc2)=O)CCCC1 C1(NC(C(CC=C)NC(C)=O)=O)CN(C(=O)Cn2ccnc2C)C(CC)(CC)C1 c1(OC)cc(F)c(S(=O)(=O)N2CCCC2(C)C)cc1F C(C(CC(C)C)NC(c1ncc[nH]1)=O)NC(C(CC)SC)=O CC(C)(CCCNC(c1sccc1Cl)=O)NC(C1CC(O)C(F)C1)=O c1(C(=O)NCC2(O)CCN(C(CC(COC)(C)C)=O)C2)cc2c(cc1Cl)OCO2 C(CO)(CCCCNC(C1CC2(C1)CC(C)C2)=O)NC(c1cc(CC)sn1)=O C1(c2n(CCN(C)C)nc(-c3ccc(CN(C)C)cc3)n2)CN2CCCC2CO1 N1(C(c2ccc(C)nc2)=O)CC(NC(=O)CCC2CCC(C)O2)C2(CCCC2)C1 C1(C(=O)NC(C2CCCCC2)C#C)CN(C)CCN1C(=O)CCC=C(C)C C1(SC)CN(C(C2CCCC2F)=O)CC1NC(=O)CCc1cc(C)no1 N1(C(C2(F)C(C)OCC2)=O)CCC2(CC1)CCN(C(C1SCCCS1)=O)CC2 N1(C(C(C)SCC)=O)CCC(F)CC1C(N1CCOC(C)(CC)C1)=O CC(C)(C)CC(O)C(=O)NC1CCC(NC(c2csc(C(F)(F)F)c2)=O)CC1 c1(C(N(C(CNC(CC(CC)CN(C)C)=O)C)C)=O)cc(C)c(C)nc1C C(=O)(C(C(C)(C)C)NC(N)=O)NCC1OCCN(C(C2C(C(N)=O)COC2)=O)C1 c1(SC)sc(C(=O)N(C2CCN(C3CCN(C)C3=O)C2)Cc2ccccc2)cc1Br CCC(C)CCC(=O)NC1(C2CN(C(c3sc(CC(C)C)nc3C)=O)C2)CC1 CC(F)(F)C(F)C(=O)NCCCC(O)C(=O)NC1CC(C)(C)C1 Cn1nc(C(N2CCC(NC(C3CCC(CO)CC3)=O)C2)=O)cc1[N+](=O)[O-].CCF C1(C(=O)NCC2CC2(F)F)C2CCC(C2)N1C(=O)CC1OCCCO1 c1(C(=O)NCCC2N(C(C3C(CC)C3)=O)CCSC2)nn(C)c2ccc(Br)cc12 Cc1cc(C(N2CCCC(NC(C3CC3C(N)=O)=O)C2C)=O)c2ccccc2n1 C(CCCC(=O)N1CCCC(NC(C2(CO)CCOC2)=O)C1)OCC C1(C(=O)NCC2N(C(C(CC(C)C)O)=O)CCOC2)C2CCC1(C)C2(C)C C12(CNC(c3c(C)nc[nH]3)=O)CCCC1CN(C(C1CC13CCC3)=O)C2 CC1CC(C(=O)NCCCn2ccnc2)N(C(c2ccccc2O)=O)C1 C1(O)(N(C(CC(C)C)=O)Cc2ccccc2)CCN(CC2CCN(CS(C)(=O)=O)C2)C1 C1(C(=O)OC)CN(C(=O)C(=O)Nc2ccccc2Br)CC1(C)C(=O)NC(C)C C1(C(N(CCC(C)C)C)=O)CC2CC2N1C(C1CC(O)CN1C)=O c1(C(=O)NCC(C(C)C)(C)NC(C2COCCOC2)=O)cccc2sncc12 N1(C(C2C(=C)CC2)=O)CC2OCC(NC(c3cn(C)c(=O)nc3O)=O)C2C1 C1(C#N)(C(=O)NCCCn2cc(-c3ccc(C)cc3)nn2)CC12CCCC2 c1(C(=O)NCCCN2CCC(NC(CC(=O)OC)=O)C2)c(C)oc(C)c1C CC1CC(NC(=O)CCc2cncn2C)CN(C(=O)CC2(C#N)CCC2)C1 N1(C(C(C)N(C)C)=O)CC2COCCC2(CNC(=O)Cc2ccccc2)C1 CCC(C)(C)C(O)C(=O)N1CC(N(C)C)C(CNC(c2cnnn2C(C)C)=O)C1 C1(N(C(CN(C)Cc2n[nH]c(=N)s2)=O)C)CCCN(C(C2CCC2)=O)CC1 c1(C(=O)NC2CCN(C(=O)Cn3ncnn3)C2)ncc2[nH]ncc2n1 Cc1cccc(Cl)c1CC(N1CC(O)(C2CCCN2C(=O)C2=CSCS2)C1)=O N1(C(c2c[nH]c(=N)o2)=O)CCS(=O)(=O)C(CCNC(=O)COC(F)F)C1 N1(C(CCC#C)=O)CC2C(F)(C1)C(c1ccccc1)NC(=O)CCC(=O)N2.CC Cc1ccccc1C=CC(N1CC2CCC2(CCNC(c2cncnc2)=O)C1)=O C12CN(CCS1)C2=O.n1(C2(CC#N)CC2)cc(C(C)(C)C)nn1.C(C)(C)(C)O C1(CNC(CN(C(C)=O)C)=O)COCCN1C(C1CC(C)(C)C1C(F)(F)F)=O CC(C)C(CCC(=O)N1CCN2CCCC2C1)NC(C1CN(C)C1)=O N1(C(Cc2n(C)cnc2)=O)CCC(c2ccccc2)(CNC(=O)C2=CCC2)CC1 c1(C(N2CCC(NC(C=CC(=O)N(C)C)=O)C2)=O)cccc(F)c1F c1(N(CC(=O)OC)Cc2ccc(CC)cc2)cnc2ccccc2c1 CC(C(=O)NC1C(C(F)(F)F)C1C(F)(F)F)C(N)c1ccccc1 C1(NC(c2ccc(C(C)(F)F)cn2)=O)CCSC12CN(C(c1scnc1Cl)=O)C2 N1(NS(NC)(=O)=O)CCC(NS(=O)(=O)C(C)C)C(C(=O)OC)C1 C1(N=[N+]=[N-])(C(=O)NC2C(OC)COC2)CCN(C(c2nc(Cl)oc2C)=O)C1 CCCCC(F)C(=O)N1CC(C2CN(C(=O)C(O)C3CC3)CCO2)C1 C(C(C)(C)C(=O)N1CCOC(C(=O)NC2CCCC2(C)C)C1)OC CCCCC(CC(=O)NC(c1[nH]c(C)nc1C)C)NC(=O)C(C)(C)Cl C1(C(N(C2CCCCC2)CC)=O)CN(C(c2ccncc2)=O)CC(C)(C)O1 C1(CN(C(c2c(C)ocn2)=O)C)CCC(NC(=O)CNC(=O)C2CC2)CC1 C1(C(N(C(C)CO)CC)=O)(NC(=O)CC(=O)OC(C)(C)C)CCC(C)(C)C1 C1(CNC(c2ccc(OC(F)F)nc2)=O)CN(C(c2n[nH]cc2C2CC2)=O)CCO1 CC(O)C(C(=O)NCC1C2CN(C(C3(N(C)C)CCOCC3)=O)CC12)N(C)C C=C1CC2(C1)CC(C(=O)NC1CCC1NC(C1CCN(CC)C1)=O)C2 Cc1ccc(OCC(=O)N(C)CC2(O)CN(C(c3cnsc3)=O)C2)cc1 N1(C(C(C)n2cccc2)=O)CCN(C(=O)CSc2cscn2)C(C2CC2)C1 C(C(CO)(CO)NC(c1cncc(C)n1)=O)N(C(C(C)(C)OCC)=O)C N1(C(CCn2ncc(C)c2)=O)CCC(NC(=O)C(F)CC2CCOC2)C(CO)C1 C1(C)(CC)CCC(C(N2CC(COC)(NC(C3CC(C#N)C3)=O)C2)=O)O1 c1(C(=O)OC)c(F)cc(NC(c2cc(Br)c(O)nc2C)=O)cc1Br n1(CCSC)nnnc1C(C1CCCC1)(C)NC1(C(C)C)CC1 c1(C(=O)NCCC(C)N(C(CCOC(C)C)=O)C)ccc(F)c(S(N)(=O)=O)c1 C(C(=O)NOC(c1ccccc1)C)(C(C)C)NC(C(CSC)C)=O c1(CC(=O)NCC2(O)CN(C(=O)Cc3cn[nH]c3)C2)csc(N2CCCC2=O)n1 CC1C(NC(=O)C=Cc2cscn2)CC2CCC1N2C(c1ccc(N)cc1)=O N1(C(C2(C)CC2)=O)CCC(NC(=O)Cc2n[nH]c(=N)s2)C(F)(F)CC1 CC1(C(=O)NCCCC(=O)OC2CCCC2)CCCN1C(=O)CC1CC1(Cl)Cl N1(C(C(C)n2cccc2)=O)CCCCC1CCNC(c1coc(Br)c1)=O c1(OC)cc(C(=O)NCC2CC3CN(C(C4(N(C)C)CCC4)=O)CC23)cc(Cl)c1 c1(C(C(=O)OC)NCc2cccc(Cl)c2OC)c[nH]c2ncccc12 CC(C)(CC(F)F)C(=O)NCC1C(Cn2cc(COCC)nn2)C1(F)F c1(CCC(=O)NC(c2cn(C3CCOCC3)nn2)CCC)ccc(C#N)cc1F c1(C(N2CC3C(CNC(c4n(CC)nnc4C)=O)(C3)C2)=O)cc(Cl)cc(C)c1C CCCCCCC(C)C(=O)NCC(CNC(=O)CCNC(=O)OC)CO c1(OC)nc(N2CCC(CCNC(=O)CC3C=CCC3)C2)nc(C)c1F CCCCC(F)(F)C(=O)NC(C)C(C)C(=O)NC1(c2nc[nH]n2)CC1 Cc1cc(C(=O)NC2CC(OCC(=O)NCC3CC4(CC4)CO3)C2)cc(C)c1 C1(NC(c2cn(C)nn2)=O)CCC(CNC(=O)CCn2cccnc2=O)CC1 C1(OC)(NCC(=O)NCC(CO)NC(=O)C(C)(C)c2cncnc2)CCCCC1 CC(C)CC(O)C(=O)NCC(C)(C)CNC(=O)C=C1CCC(C)C1 C1(CCC(=O)N(C2(CC3CC3)CC2)C)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 c1(C(=O)NC2CC(NC(C=CC)=O)C2)c(OC)ncnc1OC O=C(CC(C(F)F)c1ccc(F)cc1)NCC(O)CCNC(C1CCSCC1)=O C(=O)(C1=C(C)OCCC1)NC(CC=CC)C(=O)Nc1cn(CC)nc1C c1(CNC(CC2CCCN(C(c3c(CC)nccn3)=O)C2)=O)n[nH]c2c1CCC2 C(C(C)C(C)C(=O)NC(C)(C)CNC(c1ccc(CN(C)C)[nH]1)=O)OC Cc1nc(C(=O)N(C)C)ccc1CNC(C1CN(C(=O)C2=CCCOC2)C2CC12)=O Cc1cc(N2CCN(C(c3cnc(Cl)cn3)=O)CC2C)nc(C(C)(C)C)n1 N1(C(CC(c2c(F)cccc2F)C)=O)CCC(C)C(NC(c2csnc2Cl)=O)C1 C1(O)(C(=O)NCC2(C(=O)NCC3(C#N)CCC3)CCC2)CCCCC1 c1(C(N2CCCC(CC=C)(NC(C3COC(C)C3)=O)C2)=O)ccc(C)c(Cl)c1F N1(C(c2c(C)n[nH]c2C)=O)CCC2(CCN(C(=O)CC3CCCCC3(F)F)C2)C1 c1(NC2C(C3CCN(C(COC)=O)CC3)OCC2)ncnc2sc(C(N)=O)nc12 C1(C(C)(C)O)(CNC(CN(CC)CC)=O)CN(C(=O)CCCF)C1 C1(C(N2CCC(C(C(=O)NCCNC(=O)NC)(C)C)C2)=O)CCCC(=O)CC1 N1(C(CCOCCC)=O)CC2CCC(C(=O)NCC(=O)NOC)(C2)C1 N1(C(Cc2c(OC)c(Cl)ccc2)=O)CC(NC(=O)C=C2CC2)CC(C)(C)C1 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)C(CCOC)OC)CC(C)C1 c1(C(=O)NC(CC=C)CNC(c2csc(C(C)C)n2)=O)cc(C)c(F)cc1Cl Cc1ccc(CC(N2CCCCC2CNC(C2CCCC(C)(C)O2)=O)=O)cc1O c1(CC)nc2c(C(=O)NC(CO)CCCCNC(=O)C(C)=C3CC3)ccnc2[nH]1 N1(C(c2c(OC)nccc2)=O)CCCC(C)(CNC(C2CCS(=O)(=O)N2C)=O)C1 C1(NC(c2cnn(C)n2)=O)CCC2CCN(C(=O)C=CCCc3ccccc3)C12 N1(C(c2cnn(C(C)C)n2)=O)CCCCC(CCC(=O)NCCC(C)(C)CO)C1 C(=O)(C1CNc2ccccc21)N1CC(C2CN(C(C3(C#C)CC3)=O)C2)OCC1 N1(C(c2nn(C)c(NC(=O)C#CC(C)(C)C)c2)=O)CCC2C(C1)C2(F)F CCC(C(=O)NCCOCC(=O)NCc1ccsc1)SC N1(C(C(C=CC)O)=O)CC(OC)CC(C)C1.C12(CC=CCC1)C(=O)NC2 C1(N=c2[nH]nc(-c3ccon3)s2)(NC(c2c(N=[N+]=[N-])cccc2)=O)CCC1 N1(C(COCCC=C)=O)C(CC(=O)NC2CC2CC(C)C)C2CCCC12 C1(F)(C(=O)NC2(C(=O)OC)CC2C)CN(C(C23CCC(C2)C3)=O)C1 C1(NC(c2cc(CNC(C3C(C)C3)=O)on2)=O)CC(O)C(F)C1 c1(CC(=O)NCCC(C)NC(C2(C)CC2Br)=O)csc2ccccc12 N1(C(c2c(C)nsc2)=O)CCC2CC1CN2C(c1cc(C2CCOCC2)on1)=O CCCCC(C(=O)NCC=CBr)NC(c1cncc(NC)c1)=O C(CO)(CCCCNC(C1CC2C=CC1CC2)=O)NC(C1(C(=O)NC)CC1)=O c1(C(=O)NC(c2scc(C)n2)C(F)(F)F)ccc(C(F)(F)F)nc1 C(=O)(C(F)(F)C(O)C(C)C)N1CCN(C(c2c(C)cc(Cl)nc2)=O)C(CF)C1 Cc1c(F)ccc2[nH]c(C(=O)N(C(C)CCNC(C3CNC(=O)N3)=O)C)cc12 c1(C(=O)NC(CN(C(C2C(CCC)CCC2)=O)C)C)nc2ccccc2[nH]1 Cc1c(C(=O)NCC(C)(O)CNC(=O)COCCN(C)C)c[nH]c1C#N N1(C(Cc2c(C)scc2)=O)CCN(C)CC1C(=O)NCC(C)N(C)C C(C(CC(C)C)C(=O)NC(C)(CC(C)CC(COC(CC)CC)=O)C(F)F)NNCC c1(OC)c(CNC(c2ncccc2Br)c2nnnn2CCCF)c(C)nn1C C1(C2(NC(C(c3cnn(C)c3)C)=O)CC2)CCCN1C(=O)C(F)=CC1CC1 C1(NC(CCSCCCC)=O)C(C)CN(C(c2nc(=N)cc[nH]2)=O)CC1C N1(C(CCN(CCCCC)C)=O)CCC(F)C(NC(c2nocc2Cl)=O)C1 N1(CC(N2CCCC2)=O)CCCC(NC(CC2(C)CC2(Cl)Cl)=O)C1 C1(CC(=O)NC2CC(CNC(C3(F)C(C)C3)=O)C2)CCCCN1C C12(NC(CCNS(CC)(=O)=O)=O)CCCC1N(c1nccnc1F)CC2 C(=O)(N=S1(=O)CCC2(CCN(C(C)=O)CC2)C1)c1ccc(C(=O)OC)c(Cl)n1 N1(C(C2CC=C(C)CC2)=O)CCC2C1CCCN2C(c1ccc(Br)cn1)=O C1(C(=O)NCC(CNC(C(c2cccc(OC)c2)O)=O)C)CN2CCN1CC2C N1(C(C2CC(C#N)C2)=O)CCC2(C1)CN(C(=O)C(F)(Cl)c1ccccc1)C2 CC(O)C(F)(F)C(=O)NC1CCN(C(c2c(Cl)nn(C)c2Cl)=O)C1 CCC(C)(CC)C(=O)N1CC(C(N2CCCC2CC)=O)C(C)(C)C1 N1(C(C2CCOCC2)=O)CCCC2(CCCN2C(=O)CN2CCS(=O)CC2)C1 c1(NC(CC)CCCO)nc(C)cc(=NC2CCn3ncnc3C2)[nH]1 Cc1nc(NC(C2(F)CN(C(C3CC4(CCC4)C3)=O)C2)=O)nc(Cl)c1Br C1(C(=O)NCC(C2CC2)OCC)(C(=O)OC)CC(C)=C(C)C1 C1(CNC(=O)C=C2CCOCC2)CN(C(C2(C(F)F)CC2)=O)CC12CCOCC2 c1(OC)cc(C(=O)N(CC(C)CNC(=O)C=C(C)C2CC2)C)ccc1C#N C1(O)(CNC(CCN(C(Cc2ccn(CC)n2)=O)C2CC2)=O)CC(C)(C)C1 c1(C(=O)NCCC2(NC(C(c3ccccc3)N(C)C)=O)CC2)cnc(O)c(F)c1 N1(C(C2(CC)CCC2)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)CC12CCC2 c1(C(N(c2nn[nH]n2)C)=O)cc(O)c2sccc2c1 c1(C(=O)NC(CNC(C(C)(CO)OC)=O)(C)CO)cnn2c(C)cc(C)nc12 C1(NC(C2CN(C(C)C)C2)=O)CC2CC1N(C(=O)CCCc1csc(=N)[nH]1)C2 CN1CC(C)(NC(c2cc(Cc3ccc(F)cc3)on2)=O)CCC1=O c1(OC)c(C)cc(C(=O)N(C2CCCC2)CCCNC(=O)C2=CCOC2)cc1C c1(C(=O)NC(C2(O)CN(C(=O)C(c3cnn(C)c3)=O)C2)C)noc2c1CCCC2 C12(NC(C3(NC(C)C)CC3)=O)CCN(CC)CCC1C2.c12cc([nH]n1)C(=O)N2 CC(C)(C)CN=c1[nH]nc(-c2csc(C(F)(F)F)c2)o1 C(C)(CC(C)n1cncn1)N(C(C)(C)C)C(=O)N(N(CCC1CC1)C(C)N)C.CC C(=O)(C1=CC2(CCOC2)C1)N1C(C(=O)NC2C(O)CCN(C)C2)CCC12CC2 c1(CC(C)CC2(NC(=O)NCC(C)(C)C)CC2)cccnc1 N1(C(C(CC)Oc2cccc(C)c2)=O)CC2CN(CC(=O)NC)CC2C1 CC1C(NC(=O)Cc2cnsc2)CCCN1C(c1cnc2n1CCC2)=O C1(NC(C=CCOC)=O)CN(C(c2cccc3sccc23)=O)C2(CCOC2)C1 C1(C(=O)NC2CCC(NC(CC3CCN(C)CC3)=O)C2)CCCCC12CC2 N1(C(CC(CCC)CC)=O)C2CCC1CN(c1ncccc1[N+](=O)[O-])CC2 Cc1scc(C(=O)NC2COCC2NC(C2CCC(=O)N2C)=O)c1C C(=O)(CCCC(=O)NCC(CO)NC(=O)C(c1ccccc1F)O)OC(C)(C)C C12(NC(C(C)O)=O)CCCC1N(C(=O)C(C)S)CC2 c1(C(=O)NCCC(CNC(=O)C(C)S(N)(=O)=O)OC)cc(F)ccc1C(C)C CC1CCN(C(c2cnc[nH]2)=O)CC1NC(=O)Cn1ncn(C)c1=O N1(C(C2(OCC)CCOCC2)=O)CCC(NC(C2(Br)CC2)=O)C(F)C1 C1(C(=O)NC2C(NC(c3c(C)nn(CCO)c3C)=O)C2)CCc2ncnn2C1 N1(C(CN(C)C(N)=O)=O)CC(NC(C2CC(n3ccnc3)C2)=O)C(SC2CC2)C1 CC1CC(n2nc(-c3cc(Cl)ccn3)nc2C2CC2)CCO1 c1(C(=O)Nc2cncc(C)n2)cccc2c(-c3cc(F)cc(C#N)c3)cccc12 CC1(C)CCCCC1C(=O)Nc1ccc(C(c2ccc(F)cc2)=O)cc1F C1(C#N)(CCC=C)CCN(C(c2nnc(C)s2)C(=O)NCC2CCCO2)CC1 CC(C)(C)CCCCNC(=O)CNC(C1(Cc2nc[nH]n2)CC1)=O c1(C(=O)NC2C(C(=O)NCC3CC(OC)C3)CC2)ccc2ccoc2c1 c1(CC)ccc(NC(C2CC(F)(F)CN2C(c2ccc(C(F)F)o2)=O)=O)c(F)c1 N1(C(c2ccc(OCC=C)c(OC)c2)=O)CCCN(C(=O)CC(F)F)CC1C c1(C(=O)NCC2(C)CCCN2C(c2c(C)occ2)=O)nc2c(cc1C#N)CCOC2 O=C1CCC(CC(N2CCCCC2Cc2cn(Cc3ccccc3)nn2)=O)CN1 C(C(C(C)C)NC(=O)CC1(CCn2cncn2)CC1)NC(C(C)SCCCC)=O c1(NC(C(CNC(C2CC(OC)(OC)C2)=O)N(C)C)=O)cnc(O)n1C CC(C)CC(CCO)NC(C1CCN(C(=O)CCc2ccc[nH]2)C1C)=O C1(C(=O)NC(CCNC(C(C(C)C)SC)=O)C)Cc2c[nH]cc2S1(=O)=O C1(C(=O)OCc2c(OC)nsc2)CC2(CCC(CN)OC2)C1.C(C)(C)(C)NC(=O)O c1(C(=O)NC(C(C)C)CCN(C)C(C2CC(CF)C2)=O)cc2ccsc2n1C N1(C(C2(C)CC(C)C2)=O)CC(CNC(C2(C#N)CCC2)=O)C(O)C1 C1(C(=O)NC(CCCC)CNC(=O)C(CC)SC)CCCCS1(=O)=O C1(NC(c2ccccc2CCl)=O)CN(C(=O)C(F)CC2CC2)CCC1O Cn1ccc(CCC(=O)NC(CNC(=O)CNC(c2ccsc2)=O)C2CCC2)n1 C(c1cncc(F)c1)=CC(=O)NCC(CNC(C(CC)(F)F)=O)C C1(C(=O)NCC2CC(NC(C3(C)CC3)=O)C2)COc2ccc(Cl)cc2C1 c1(C(c2ccco2)=O)ccc2c(c1)NC(C)C2.Cc1ccc2cc1N(CCO)C2=O c1(NC2(C(F)(F)F)C(F)(F)C2)nc2cc[nH]c2c(=NCCn2cncn2)[nH]1 c1(OC)ccccc1N(C)C(C1(O)CCN(C(=O)Cc2ccccc2)C1)=O c1(C(=O)NCC2N(c3nccc(C)n3)CCC2)c(Cl)ccc2c1OCO2 c1(C(=O)NC2(CO)CCN(C(C3CCO3)=O)C2)cnn2c(=O)cc[nH]c12 Nc1cc(Cl)ncc1C(N1CC(CNC(=O)CCn2cccnc2=O)C(O)C1)=O C(CC(=O)NCc1cncc(C#N)c1)(C(F)F)NC(C1(C)N(C)CCC1)=O c1(C(N2C(C)CC(NC(CSC(C)C)=O)C2)=O)ccc2ccn(CC(F)F)c2c1 C(=O)(CC(C)CN(C)C)NC(CO)C(C)SC.C(=O)(CC1(NC=O)CC1)OC C1(NC(CC(=O)OC)=O)CC2CN(C(=O)CC3CC(=O)NC(=O)C3)CCN2C1=O c1(C(C(C)Nc2ncccc2-c2ccncc2)=O)cc2ccccc2s1 Cc1ccn(CC(N2CCC(CNC(c3c[nH]nc3-c3cnn(C)c3)=O)C2)=O)n1 Cc1cc(N2CCN(CCNC(=O)C(c3ccccc3)C)CC2)c(F)cc1[N+](=O)[O-] c1(C(N(CCNC(=O)CC2CCC(O)C2)CC)=O)nnn2c1CCCCC2 c1(C(N2CC3C(CNC(Cc4c(C)noc4)=O)(C3)C2)=O)cnc2ncc(Cl)cn12 C(=O)(CC(C(C)(C)C)NC(=O)CN(C1CCC1)C)NCc1c(C)nc(C)n1C C1(NC(c2n(CCC)nc(C)c2)=O)CCN(C(=O)CC2(CO)CCC2)CC1(C)C C1(C(=O)NCCC(CC)C)CC2CN(C(=O)C(O)CCSC)CC2C1 n1(C(CC)C)ccc(=NC(=O)C2CCCCCC2NC(=O)COC)[nH]1 c1(OCC)ncc(C(N2CC3CC3(CNC(C34CCC(C3)OC4)=O)C2)=O)cc1Cl c1(C(C)C(=O)N(C)CC2COCCN2C(=O)CO)ccc(Br)cc1F c1(CC)c[nH]c(C(=O)NCCC2CC(NC(=O)CCc3ccn(C)n3)C2)c1 CC(O)CC(C)CN=c1[nH]c(=NCC2(n3cc(Br)cn3)CC(CO)C2)[nH]c2cc[nH]c12 N1(C(C(C)(C)N2CCCC2)=O)CCCCCC1CO.N12CC3(CC3(CO)C1)C2=O c1(C(N2CCN(C(C(CC)n3nccc3C)=O)CC2)=O)c(F)cc(Cl)cc1Cl C1(O)(C(=O)NC2CCC(NC(Cc3c(C)ccnc3)=O)CC2)CCC(C)(C)CC1 C1(NC(=O)Nc2ccc(F)nc2)C2CC(NC(c3coc(C(F)F)c3)=O)CC12 Cc1ccc(-n2cc(C(C)NC(c3cncc(F)c3Cl)=O)nn2)c(F)c1 c1(C(=O)NCC2CC(O)(CNC(C3(CC)CCCC3)=O)C2)cnc(Cl)cc1N CC1(C)CC(CNC(C2CCC2)=O)CN1C(c1csc(-c2cccc(Cl)c2)n1)=O C1(C(N2CCCC2c2cn(CCCCCCO)nn2)=O)CC(c2ccccc2F)=NO1 N1(C(C2CC(C)(NC(c3nn(CC)nc3C)=O)C2)=O)CCn2nc(C)cc2C1 c1(OC)cc(OC)c(C(=O)NC2C=CC(C(=O)NCCS(=O)(=O)N(C)C)C2)cc1Cl C1(CNC(C(CC=C)CC)=O)CC(O)C(O)CC1C(=O)NC1(c2ccncc2)CC1 C12(C(=O)NC(C(C)NC(c3cscc3Br)=O)C)CC3CC(CC(C3)C1)C2 C#CC1CN(C(=O)C(C)C(O)C(C)C)CCN1C(=O)CC1CCCN(C)C1 N1(C(C(CC)N(C)C)=O)CC2CC1CN(C(=O)CCNC(=O)OC(C)(C)C)C2 N1(C(C(C)OCC)=O)CCC2(CCCN2C(C23CCC(CC2)C3(C)C)=O)C1 CCC(CC(=O)NC1(C(N2CCC23CC(O)C3)=O)CC1(C)C)C(C)C C1(C(N(C2CCN(C(=O)Cc3cc[nH]n3)CC2)CCOC)=O)CCS(=O)(=O)CC1 C(=O)(C1CCCn2ccnc21)N1CC=CC(NC(c2nn(C)c(Cl)c2Cl)=O)C1 N1(C(COCCC=C)=O)CC(CNC(=O)Cc2cccc(C)c2)OC(C)(C)C1 C1(NC(=O)OC(C)(C)C)CC2CCC(C1)C2(C)NC(c1ccc(CC2CC2)s1)=O C1(O)(C(=O)NC(C)CNC(C2CC2(F)F)=O)CCCC(C)(C)CC1 c1(NC(N)=O)ccc(C(=O)NC2CCCC2NC(c2cnnn2C2CC2)=O)cc1 c1(N(CCCS(N)(=O)=O)C)ccc(S(=O)(=O)NCc2cccnc2)cc1C#N C(=O)(C(C)(C)CCC#N)NC1C(CNC(c2c(C)nc(C3CCCO3)s2)=O)C1 C1(C)(C(=O)NCC(CC=C)NC(=O)C(=O)Nc2cccc(C)c2)CCNC1=O N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCn2c(CNC(C3(F)CC3C)=O)nnc2C1 C1(NC(c2cn(CC)nc2)=O)CN(C(C2CCO2)=O)CCC1(C)C N1(C(=O)COCC2CC2)CCN(C(=O)CCc2cscn2)C(CCO)C1 C1(C(=O)NCC2N(C(C3C(C4C(C)C4)C3)=O)CCC2)CCCS(=O)(=O)C1 CCCCCC(F)C(=O)NCCn1cnc(C(=O)NC2CCC(F)CC2)c1 N1(C(C2(C3N(C(c4n(CC)nc(C)c4)=O)CCC3)CC2)=O)CCCSCC1C n1(CCNC(C(C)NC(=O)OC)=O)cc(C(=O)NC(C2CCOCC2)(C)C)nn1 N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCC1C(NC(c1c[nH]nc1C(F)F)=O)C2 c1(OC)ccc2c(c1)C(C)(C)N(c1cncc(OCOc3ccccc3)n1)CC2 N1(C(C2(COC)CC2)=O)CCC2(CCN(C(C3CC4CC3CC4(F)F)=O)C2)C1 C(=O)(CCC(F)(F)F)N(CCC(C)NC(=O)CCOC(C1CCCO1)CCC)C N1(C(C2=CCCN(S(c3c(C)onc3)(=O)=O)C2)=O)CCc2nc(Br)sc2C1 C(CCC(C)C)(C(=O)NCC(C)(O)C1CCC1)NC(c1c(C)scc1)=O C(=O)(CCC(=O)N(C1CCOC(CNC(C)=O)C1)C)NC N1(C(CC(COC)C)=O)CCC(NC(c2cc(OC(C)C)ccc2N)=O)C(F)C1 CON1CCC(CC(N2CCCCC2(C)C(N)=O)=O)CC1 N1(C(c2cc(C)sc2C)=O)CC2(CO)CC1(C(N1CCCC(C)(F)C1)=O)C2 C12(CNC(c3c(N)nccc3)=O)CCC1CCN2C(C1(CCO)CC1)=O C1(C(=O)NCc2cccc(NC(C(CSC)OC)=O)n2)CCCN(C(C)=O)C1 CC(C(=O)NC(Cc1cn(CC2(C(C)(F)F)CC2)nn1)CC(=O)O)C(C)(C)C c1(C(=O)NC2C(NC(=O)CCF)CCOC2)ccc(Br)c(O)c1 c1(C(CNC(=O)CC2CC2C(C)C)NC(C=C(C)C(C)C)=O)ccc(C#N)cc1 CC1CCN(C(C2CNC(=O)N2C)=O)C(C)C1NC(=O)Cc1ccoc1 C1(NC(C2CC(C)OC2)=O)(CNC(=O)OC(C)(C)C)CCCCC1C c1(NC(=O)OC)cccc(NC(=O)CC(C)C2CCCO2)c1 N1(C(C2(CC=C)CCCC2)=O)CCC(O)C(NC(c2cnn(C)c2C)=O)C1 c1(C(N2CCC(NC(C(C)CF)=O)C(O)C2)=O)c(F)ccc(O)c1O n1(CCC)ccc(C(=O)NC(C)(C)CC=CC(=O)N(C)CC2COCCO2)n1 Cc1cocc1C(=O)NC1(C(N2CCC(NC(N)=O)C2)=O)CC(F)C1 C1(C)(CN=C(NC(C2(C)CS(=O)(=O)C2)C)NC2CC2)CCC(C)(C)CC1 C=CCC(CC=C)C(=O)N1CCC2C(NC(C3CC(OC)C(OC)C3)=O)CC12 CC(C)CC(C)(CNC(C1CC2CC1CC2O)=O)NC(=O)Cn1ncn(C)c1=O c1(CNC(=O)NC2CC(F)(F)C2)ccc(N(C2CCCC2)C(N)=O)c(F)c1 N1(C(c2cc(OC)ncn2)=O)CC(C)(C)CC1CC(=O)NC(C1CCOC1)CO C(CCCCC(=O)NC1CCC(NC(c2cc(C3CC3)[nH]n2)=O)CC1)=CCCC C12(C(=O)NC(CCCCNC(C(C)=C3CCCC3)=O)C)CCC(C)(C1)OC2 c1(OC)ccc(F)cc1C=CC(N1CC(CC(C)NC(=O)C(C(C)C)OC)C1)=O C=CCC(C(=O)NCCOCCN(C)C(C1CN(CC2CCCC2)C1)=O)C(C)C C1(OC)(CNC(=O)CC23COC(C)(C2)C3)CCN(C(=O)Cc2ccc(Cl)nc2)C1 C1(C(N2CCC(N(C(=O)C=CC3CCOC3)C)CC2)=O)(CC)CCCCC1 N1(C(C=NOC)=O)CC2CCCCC2(NC(C2CC(=O)NC(=O)C2)=O)C1 N1(C(CC(C)OC)=O)CC2N(C(c3nn4cccnc4c3Cl)=O)CCC2(C)C1 S(=O)(=O)(c1ccc(C#N)c(C(=O)OC(C)C)c1)NCc1scc(CC)n1 CC(CCCc1ccccc1)C(=O)N(C)CC1CCCCC1 S(=O)(=O)(c1cccc(NC(C2(n3cccn3)CC2)=O)c1)Nc1cc(C)on1 c1(S)cc(F)cnc1Br.n1(CC)c(N(C)C)nnc1CO Cc1ccc(CC(N2CC(NC(c3c(C)coc3C)=O)C(O)C2)=O)cc1C c1(C(N(C2CC(NC(C3(OC(C)=O)CC3)=O)C2)C)=O)csc(-c2cnn(C)c2)n1 N1(C(c2c(C(C)C)noc2)=O)CCC(NC(=O)C(C)(C)c2ncco2)C(F)C1 CCCC(CC)C(=O)N1CC(CC(=O)NCC2SCCS2)CC1(C)C CCCCC(O)CC(=O)NC1CC(CCNC(C2CC2c2ccc(C)cc2)=O)C1 C1(CC)CCCC1(C)C(=O)NC1CC(NC(c2conc2C(F)(F)F)=O)CC1O C=C(Cl)CC(C(=O)NCCCSC(F)F)NC(=O)CC1CC12CC2 C(=O)(C1=C(F)CN(C(C2C=C(C)CS2)=O)CC1)NCCC(CCC)C1CC1 C(CCCCC(=O)N)N(C(C(C)OCC=C)=O)C.C(C(C)(C)N1CCCC1)OC(F)F N1(C(C(CC)SC)=O)CC2(CNC(c3coc(C(F)F)n3)=O)CC2(C(F)(F)F)C1 Cc1c(F)ccc(C(=O)NCC2CCC2NC(C2(C)CCCS2(=O)=O)=O)c1F C(CC(Cl)=CC(=O)NCCCN(C(c1cocn1)=O)CC1CCCC1)N(C)C N1(C(CNC(C)=O)=O)CCCC(C2CC2NC(c2scc3c2OCCO3)=O)C1 C1(NC(C=C(C)C(C)(C)C)=O)CCN(C(C2CC3(CC3)CO2)=O)C12CC2 c1(C(N2CC(C)(NC(C3CC3(C)C)=O)C2)=O)ccc(Cl)c(S(N)(=O)=O)c1 c1(OC)ccc(CC(C)Nc2cccc(N(C)C)c2)cn1 c1(C(N(C(C)C)C)=O)sc2ncccc2c1Cl.C12CC(F)CN1C(=O)OC2=O S(=O)(=O)(c1cccnc1N1CCCC(F)C1)N(CC(C)O)Cc1ccc(C)o1 C(=O)(CC(C=C)CCC)NC(C(=O)NCC(C#C)CC1CC1)Cn1cncn1 c1(CNC(CCNC(c2nc(CC)oc2)=O)=O)ccc(O)cc1 CCCC(C)(CC)C(=O)NC1CCCN(C(c2noc3ncccc23)=O)CC1 N1(C(C(C2CCN(C(CN(CCOC)C)=O)C2)C)=O)CCCC1(C)C c1(C(=O)NC2C(NC(C(CC)NC(N)=O)=O)COC2)cn2cccc(Cl)c2n1 Cc1cc(CN=C(NCC2CC3CC2C3)NC(C2CCCO2)C)cnc1F CC1CN(Cc2cccs2)CCN1C(c1ccc(C(F)(F)F)nc1Cl)=O C1(N(C(=O)CCC(=O)N(C)C)CC)CCN(C(C2CC(O)C2)=O)CCC1(F)F n1(CC)cc(S(=O)(=O)N2CCCC(CNC(c3ocnc3C)=O)C2)cn1 C1(NC(N2CC(n3ncc(C(=O)OCC)n3)C2)=O)CCC2(CCC2)OC1 CCCC(C)(CC)C(=O)N1CCOC(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 N1(C(c2c(OC)n(C)nc2C)=O)CCCC2(CCN(C(=O)CC3CSC3)C2)C1 c1(C(=O)OCC)cc2c(cc1NC(c1cc(C)cc(I)c1)=O)OCO2 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CC(O)C1C2NC(C1CCC(=O)O1)=O C1(NC(CC(=C=C)C)=O)CC2COCC(C1)N2C(=O)C(C)OC1CCOC1 c1(CC)ncc(-c2cn(C3COCC3NC(=O)C(COC)N(C)C)nn2)o1 N1(C(C(c2cccnc2)=O)=O)CCC2(CCCN(C(C3CCCSS3)=O)C2)C1 N1(CC(N2CCC(C3CCCCO3)C2)=O)CCC(F)CC1 N1(C(c2ccc(CC)cc2N)=O)CCC2(CC1)CC2NC(=O)C(C)(C1CC1)OC C1(C(=O)NCC2OCCCN(C(CNC=O)=O)C2)CCC2(CCOCC2)O1 c1(CC)cc(NCC2C3CN(C(c4ccc(OC)cc4F)=O)CC23)cc(F)c1 CC1(O)CCCN(C(C2CCC(CNC(c3cc(F)ncc3Br)=O)CC2)=O)C1 N1(C(c2ccc(OC)s2)=O)CCC(NC(=O)CCSc2ccccn2)C(C)C1 CC1CCN(C(C23CCC(CC2)C3)=O)CC1CC(=O)Nc1cccc(C(F)F)c1 C1(C(=O)NC(CCC)CO)CN(C(C2CN(C(C)=O)C2)=O)CC(C)(C)C1 C(=O)(CCC(C)(F)F)NC1CCN(C(Cc2c(C)ocn2)=O)C1 c1(C(=O)NCC2CCN2C(=O)COC(F)F)cc2oc(Br)cc2[nH]1 O=C1CC(C(=O)N2CCCCC(CNC(=O)C(C)(C)N3CCCCC3)C2)=NN1 c1(C(=O)Nc2ccc(-c3cccn(C)c3=O)s2)n[nH]c2c(F)cccc12 c1(NCC(=O)NCC(C)NC(=O)CCCc2cnccn2)ccc(C(N)=O)cn1 c1(CNC(NCC2CCCC(OC)C2)=NCCN2CCC2)n[nH]c2ccccc12 C(N=c1[nH]cnc(Cl)c1NC)C1OCC(CNC(c2nc(C(=O)OC)cs2)=O)C1 c1(CC)cc(C(=O)NC(CNC(c2c(OC)cccc2Br)=O)CC)cc(O)n1 c1(C(C(=O)NCC=C)N(C2CCC(C)C2)C)ccc(C)c(I)c1 C(=O)(C1CCCn2cnnc21)NCCN1CCN(C(C2ON=C(CC)C2)=O)CC1 CON1CCC(C(N2CC(C)(C)CC2C(=O)NC2(CCF)CCC2)=O)CC1 C1(CNC(C(CC)(C)C)=O)(NC(=O)CCCc2cnn[nH]2)CC2CCC1C2 C(=O)(CCC(C)(C)C)N(C1CCN(C(CCCCNC(C)=O)=O)CC1)C c1(C(c2n(CC(=C)C)nnn2)NCC2C=CCC2)ccc(-c2nnco2)cc1 c1(CNC(C(N2CC(S(C)(=O)=O)C2)c2c(Br)cn(C)n2)=O)ccc(F)cc1Cl c1(C(=O)NC(CN(C(=O)Cc2nonc2C)CC)C)cncc(NC(C)C)n1 C(CC1CC1)(CC(=O)N(C)C(c1cnn(C)c1)C)NC(C1(C(=O)NC)CC1)=O N1(C(CCCOCC)=O)CCC2CN(C(=O)CN=S(C)(C)=O)CCC2C1 C#CCC(O)C(=O)NC1(CCC(=O)NCCSCc2cccnc2)CCC1 c1(C(N2CC(NC(C34CCC(OC)C3C4)=O)CC2(C)C)=O)ccc2c(c1)NCC2 Cc1cc(NC(C2CCCN(C(c3cc[nH]n3)=O)C2)=O)cc(C)c1F O=C(C1=CC(O)C(O)C(O)C1)N1CCCN(Cc2ccc(O)c(CO)c2)CC1 C1(CC(=O)NCc2ccc(C(=O)NC(CSC)(C)C)o2)CCC(C)CO1 C(C)(C)(CC(F)C(=O)N1CC(C)CC(O)C1)NC(C(CC=C)CC)=O N1(C(=O)OC(C)(C)C)CC2(CCC2)CC1CNC(C1CCC(N=[N+]=[N-])C1)=O c1(NC(C=CC2C(=O)NC2)=O)ccc(NC(=O)NCCCl)c2cccnc12 C(=O)(CCCN=[N+]=[N-])N1CCCC(CN(C)C(c2ncsc2Br)=O)C1 C[Si](C)(C)c1ccc(-c2csc(NC(=O)CC3(O)CCC3)c2)cc1 C(=O)(C1=COCCO1)N(C1CCCCC1)CCNC(c1cc(C(C)C)n(C)n1)=O c1(C(N2C(CNC(CCOC(C)=O)=O)CCCC2)=O)cc(C)c(S(N)(=O)=O)cn1 C1(C(N2CC(OCCNC(=O)CCC3CCCCC3)C2)=O)CC2(C1)CC(F)C2 N1(C(=O)COCC2CC2)CCC2CN(Cc3ccccc3)CC12 CCCC(CCCNC(=O)CC1CCCC(C)(C)C1)NC(c1c[nH]nc1C1CC1)=O Cc1ccc(C=CC(=O)N(C2CCC(NC(=O)Cc3ccoc3)C2)C)o1 Cn1cc2cc(C(=O)NC3CC(O)CN(C(=O)C4=NOCC4)C3)ccc2n1 C(c1cnc(O)nc1O)=CC(N1C(C)C(NC(c2nn[nH]c2Cl)=O)CC1)=O Cn1c(I)cc2c(N(C3CCCNCC3)Cc3cncc(F)c3)ncnc12 CCCCC(=O)C(=O)NCC(O)C(=O)NCc1noc(C)n1 Cc1cc(NC(=O)Cc2nc(-c3ccccc3)ns2)cnc1O N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC2(C1)CN(C(=O)COC(=O)CO)C2 Cc1cc(C(C)C(=O)NC23CC(NC(=O)CC4CSCCS4)(C2)C3)cc(C)c1 C1(NC2CCN(C(=O)OC)C2)CC=CCC1C(=O)OCC1=C(C)CCC1 C(C(=O)NOCCF)(C1CCCC1)NC(c1cc(CC)sn1)=O C1(C(C2CC2)NC(C(=O)N(C)C)=O)CCC(C(=O)NC2(C)CC(O)C2)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(=O)NCC2CC2)ccc(F)c(F)c1 c1(CNC(C(CC#C)NC(=O)Cc2cnc(C)s2)=O)ccc(F)c(C)c1 CC1CCC2(CC1)CCC(COC(c1nn(C)c3c1CCCC3)=O)O2 C1(CNC(Cn2c(C)nnn2)=O)CCC2(CCN(C(=O)CNC=O)CC2)O1 C1(CC=C)(C(=O)OCC)CCCCN1C(=O)Cn1cc(-c2ccc(Cl)nc2)nn1 C1(CC(=O)NCC2(CO)CC3(CC(C)(C)C3)C2)C(=O)Nc2ccccc2S1(=O)=O CC(C)CC(C)CC(=O)N1CCC1CNC(c1cc(=N)[nH]cc1Br)=O C1(NC(CN2C(C)CCC2C)=O)CC2CCC(C1C)N2C(c1ccnn1C)=O N1(C(C2(CC)CCN(C(=O)Cn3cncn3)C2)=O)Cc2ccccc2C1 Cc1cccnc1CCC(=O)NCCC1CCC(NC(=O)Cc2csc(S)n2)C1 C1(C(=O)NCCC(C)NC(=O)Cc2cnsc2)CCC(=O)N(CC(F)(F)F)C1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CC(CNC(=O)C(C)OCC(C)C)CC1(C)C N1(C(c2ncn(C)c2)=O)CC2CCC1(CNC(C1(C)CCC(F)(F)C1)=O)CC2 C(=O)(C(CC(=O)OC(C)(C)C)NC(C)=O)N1CCC(C(CNC(C)=O)F)CC1 C1(NC(c2c(CC)oc(C)c2)=O)CC2(C1)CC(C(=O)NC1(CC)CC1)C2 C(CN=c1[nH]nc(CC(C)C)s1)N.C(c1nc(C)co1)=CC(=O)N(CC)CC N1(C(Cc2scc(C)c2)=O)CCCC(C2CN(C(=O)CC3=NNC(=O)C3)C2)C1 N1(C(C2(F)CCN(C(c3c(C)ncs3)=O)C2)=O)CCC2C(O)C(C)(C)C12 C1(NC(=O)CC2CCCCC2F)Cc2ccccc2C1NC(c1ccoc1Br)=O N1(C(CCCC#C)=O)CCCCC12CC(NC(=O)CC1(CSC)CC1)C2 N1(C(C(C(C)C)SC)=O)CCC2(CCN(C(c3cc[n+]([O-])cc3)=O)C2)C1 CN1CC(C)(NC(C2(F)CCN(C(C3CCC=CCCC3)=O)CC2)=O)CCC1=O c1(CNC(C2(CNC(C3C(CC)CCC3)=O)CCC2)=O)cc(C)c(C)o1 c1(C(=O)N(Cc2ccccc2)CC2CCCCC2)cc(Br)c(O)cc1F c1(C(=O)NCCNC(c2cccc(-n3cncn3)n2)=O)cncc(O)c1 c1(OCC(=O)NC2CCC(N(C(=O)CCN3CCC3)C)C2)ccc(F)cc1F c1(C(N(CCCNC(C(CC)C(C)C)=O)C2CC2)=O)cc(F)c(OC)c(Cl)c1 C1(C(=O)NC2(C)CCN(C(c3c(CC)nn[nH]3)=O)C2)Cc2nccnc2C1 N1(CC(=O)NC(CC(C)NC(C=CC=CCC)=O)C)C(=O)c2cccnc2C1=O C=Cn1nccc1C(=O)N(CCC(=O)NCC(N1CCCC1)=O)C N#CC1(CC(=O)NC2CC(F)CN(C(=O)CSCc3ncc[nH]3)C2)CCCCC1 C(=O)(C1=CCC(C)(C)CC1)NCC(C)CNC(=O)COC(C)(C)C CC1CN(c2ccc(C(N3CCC(O)(c4ccc(F)cc4)C3)=O)cc2)CCN1 N1(C(Cn2c(C)ncc2)=O)CCC2(CC1)CC2C(=O)NCc1ccc(F)cc1F c1(C(N2CCN(C(c3n(C)cnn3)=O)C3C2C3)=O)ccc(C#N)c(F)c1 N1(C(C)=O)CCCCC1CCC(=O)NCCCNC(c1ccnn1CCF)=O C#CCCCC(=O)NC(c1ccccc1)C(=O)NCC(c1cccnc1)O C12(C(=O)OCC)CN(CCC(N)=O)CC(CO)(C1)C2 c1(NC(c2ccccc2-c2cc(F)c(F)cc2Cl)=O)cc(F)c(Br)cc1Br C(=O)(C(CC1CC1)NC(=O)Cn1cnnn1)NCC(C)(O)C(F)F C1(NC(C2CC2CC(F)F)=O)CCCC1Cc1ccccc1 C1(C(=O)NC2CC(CNC(c3c(C)n[nH]c3)=O)C2)CCC2(CC1)NC(=O)NC2=O N1(C(CCCC2C(C)C2)=O)CCC(CC(=O)NC(C)CC(=O)N(C)C)C1(C)C C(=O)(C1=NOC2COCC12)NC1CC2CC(NC(C3C(CC)C3)=O)CC21 c1(CC(C(=C)C)OC)cccc(NC2CCCCC2C)c1 c1(C(CC)OCCNC(=O)CSCC(C)C(=O)O)cc(C)ccc1C Cc1noc2ncc(C(=O)NC(C)CNC(C3(F)CCOC3)=O)cc12 C(=O)(C(CCNC(c1cc(C(C)C)on1)=O)OC)NCCc1cn(CC)nc1 C12(C(=O)NC(CN(C(=O)Cc3c(C)n[nH]c3C)CC)C)CCCC1(C(N)=O)C2 c1(C(N(CC)Cc2csc(Cl)c2Cl)=O)cc(C)ccc1CN1CCCC1 C1(CC(=O)NCC2(O)CN(C(C3COC(=O)O3)=O)C2)CC2C=CC1C2 Cc1cnc(C(=O)NCCC2CSCCN2c2ncnc(=N)[nH]2)c(C)c1 C(=O)(C(F)C(=O)NCC1(C(=O)NC2(C)CC(O)C2)CC(C)(C)C1)OCC N1(C(c2cc(CC)sn2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)CC(C)C1 C1(NC2CC(C(C)NC(C3C(c4cn(C(C)C)nc4)C3)=O)C2)CCCCCCC1 c1(-c2cc(C(=O)NC3C(NC(Cc4cc(C)on4)=O)CC3)no2)ccc(C)c(C)c1 N1(C(c2ccc(OC)c(C)c2)=O)CCC(OC(C)C)CC12CC2 N1(C(C2N(CC)CCOC2)=O)CCC(F)(CNC(c2cn(C)cn2)=O)CC1 C1(NC(COCC#C)=O)CN(C(=O)CCN2C(C)CCCC2C)C2CCCC12 CC1(CNC(=O)CC2CCC(O)C2)CCCN(C(C2CCC2)=O)C1 c1(SC)ccc(C)c(C(=O)NCC(CO)NC(=O)CC#N)c1 C(=O)(CCC(C)OC)N(CC(C(N1CC(C)(CC=C)C1)=O)C)C C=C(C)CN=C(NCC(C)CN1CCC(C)CC1)NC1CC(N2CCCC2=O)C1 N1(C2CN(C(=O)OC(C)(C)C)C2)CC(C(=O)Nc2cncnc2C)NC1=O N1(CC)C(=O)CCC1Cc1cn(C2CCCN2C(c2nccn2C(C)C)=O)nn1 C1(C#N)(C(=O)OC(C)C(=O)N2CCCC2)CCOC1.c12ncoc1C(=O)N2 C1(C(=O)NC2CCC(OC)C2)CCCN(C(C2(CC3CC3)CC2)=O)CC1 C(N=c1cc(NCc2ocnc2C)nc[nH]1)C1(CC)CCC1 C1(NC(c2ccc(-n3c(C)cnn3)cc2)C2CC2)CCNCCC1c1ccccc1 N1(C(C(C2CN(C(=O)CC3CCCOC3)C2)O)=O)CCCC12CCOC2 C(CCCN=c1[nH]c(=NCCC(C)N(C)C)c2sccc2[nH]1)N(CC)CC c1(C(C(=O)NCC(CNC(C(C)SCCCC)=O)(C)C)F)ccc(F)cc1F c1(C(N2CCCC(CC(=O)NCCC(=O)OC(C)C)C2)=O)cc2c(s1)CCC2 c1(NC(C2CS(=O)C2)=O)c(F)cc(Cl)cc1Br S(=O)(=O)(CC(=O)N(C1CCCC(NC(=O)Cn2ccc(C)n2)C1)C)N(CC)CC C(=O)(CC(C(F)F)NC(C1C(C)C1C)=O)NCC(C(=O)NC)(C)C N1(C(C(C2CCOCC2)OC)=O)CC(C)(C)CC1CNC(C1(O)CCCCC1)=O N1(C(CCc2n(C)ccn2)=O)CCOC(CCCNC(=O)C=CC2(C)COC2)C1 CC1CC2CCC(C(N3CCN(C(C4COC(C)C4)=O)CC(C)(C)C3)=O)CN2C1 CCC(C#N)C(=O)N1CC(F)CC1C(=O)Nc1cnn(C(C)C)c1 Cc1c(C(=O)N(C)CC2COCCN2C(C2CCOC2)=O)cccc1Br N1(C(C(CC)NC(C)=O)=O)CC2CCC(CNC(C3CCCCC3)=O)C2C1 CC(CC#N)C(=O)NCCn1cc(CNC(=O)CC(C)(C)C)nn1 c1(C(N(CCCOCCN(C(=O)CCCSC(C)(C)C)C)C)=O)ccc(Cl)cc1 c1(OC)cc(OC)cc(C(=O)Nc2ccc(-c3cn(CCO)nn3)c(C)c2)c1 C1(CNC(c2ccc(NC)cn2)=O)COCCN(C(c2c(C)nsc2C)=O)C1 C1(NC(c2c(CC)n(CC)nc2)=O)CCCN(C(=O)CC(=O)OC(C)(C)C)C1C C12(CC#C)CCC1CN(CC(=O)NCCNC(=O)C1CC1)C2 Cc1nc(C(=O)NCC2CC(NC(c3csc(C(N)=O)n3)=O)C(O)C2)cc(O)n1 CC1(C)CC(CNC(=O)CN2CC3CC3C2)N(C(=O)CC2CC(O)C23CCC3)C1 C1(NC(N2C(CC(N)=O)CCCC2)=O)CC(F)(F)C12CCC2 c1(OCC#C)ccc(COC(c2cscc2C(F)F)=O)cc1 C1(NC(Cn2c(C)ccn2)=O)CC2CCC(C1C)N2C(c1cnc(C2CC2)s1)=O N1(C(c2ccc(C(C)=O)[nH]2)=O)CCCOC(CNC(=O)CC23CCCC2C3)C1 CC(C)C(C(=O)N1CC(OCC(=O)NC(C(F)F)C(F)(F)F)C1)NC(=O)N(C)C CN1CCC(C)(C(=O)NC(C(=O)Nc2ccc(N(C)C)nc2)c2ccco2)C1 CN1N=C(C(=O)NCC2OCCC2NC(C2CC(CO)N(C)C2)=O)CCC1=O CC(C)C(CNC(=O)CCc1cnccn1)C(=O)NC(CN1CCCC1)CO S(=O)(=O)(c1cccnc1NC1CCCC2(CC1)CC2)NCC12C(C)(C)C(CC1)C2 C12(C(=O)NCCN(C(c3ccnnc3S)=O)CC)CC(C1)C(C(F)(F)F)O2 C1(CC(=O)NCC2(CCNC(CCNC(N)=O)=O)CCC2)CNC(=O)O1 c1(CNC(C(C2CCC2)OCC)=O)nc2c(s1)CN(C(c1[nH]cnc1C)=O)CC2 Cc1cc(NC(c2nnnn2CCCF)CCC2CCCC2)cc(Cl)c1 Cc1cc(Cl)c(C(=O)NC2CCN(C(=O)C=Cc3ccncc3)CC2CO)cn1 Nc1cc(C(=O)NC2CCCC2NC(c2cncc(C(F)(F)F)c2)=O)cc(Cl)n1 c1(C(=O)NCCC(C)(C)CNC(=O)CCc2nncs2)ncsc1S(N)(=O)=O CC(Cc1cn(C(C)C(=O)NC23CC(C(=O)N(C)C)(C2)C3)nn1)C(=O)O N1(C(c2c(C)cco2)=O)CC2(C1)CN(C(C1CC1C1CC1C)=O)CCO2 c1(NC(=O)Nc2c(N(C)C)cccc2)cc2c(cc1Cl)NC(=O)C2 Cc1ccc(Br)c(C(=O)NC2CC23CC(NC(=O)Cc2cnc[nH]2)C3)c1 c1(NC(N2CCC(C)(CC(=O)OC)CC2)=O)cc(Cl)c(Cl)cc1SC N1(C(CC(C=C)C)=O)CC2CCC(C1CO)N2C(c1ccc(C)cc1C)=O C1(C(=O)NCC2(CNC(C3(F)CCC3)=O)CC2(F)F)CC12CCSCC2 C1(N(C(=O)COCc2ccncc2)C)CCC2CN(C(=O)C(C)(C)C)CC12 C#CCC(CC#C)C(=O)NC(CN(C)C(c1cccc(OC)n1)=O)CC c1(C(=O)NCC2(C)COCCN(CCNS(C)(=O)=O)C2)ccc2oc(O)nc2c1 C1(C(N2CC(CN(C)C(c3cnnc(O)c3)=O)C2)=O)(CC)CCCCC1 C1(NC(CN(C)C(=O)C2CC2)=O)CCCN(C(C2CC3(CC(=O)C3)C2)=O)CC1 C(=O)(C1=CCC(NC(C2(SC)CC(=O)C2)=O)C1)NCCCC(=O)NC c1(C(=O)NCC(CC)NC(=O)C=CCN(c2ccco2)C)ccc(F)c(C2CC2)c1 c1(NC)cncc(C(=O)NC2CCCCC2NC(c2csnc2C)=O)n1 C(=O)(C1=CCCCC1P(C)(C)=O)NC12C(CN(C(c3c(C)cc(F)s3)=O)C1)C2 C1(NC(c2nn(C(C)C)c(C(F)F)c2)=O)CN(C(=O)CSC2CC2)CCC1C C1(C(=O)NCC2C(C)CN(C(=O)C#CC3CCCC3)C2)CCC(C2CCCO2)O1 C1(N(C)C(c2conc2-c2ccccc2)=O)CCCN(C(=O)CC2CCOC2)C1 c1(CC=C)ccc(OC)c(NC(C2CCN(C(C3CC3C(C)C)=O)CC2O)=O)c1 C1(C)(C(N2CC(C)C(NC(C3(C(F)(F)F)CCCC3)=O)C2)=O)CC2(CCC2)C1 C1(C(=O)NCC2(O)CN(C(c3c(CC)oc(C)c3)=O)C2)CCC2(CCC2)O1 CC(C)CCC=CC(=O)NCCCN(C(C1COC(C)C1)=O)Cc1cccnc1 C1(NC(c2n(C)ncc2Cl)=O)CN(C(=O)Cc2ccn(C(F)F)n2)C2(CCC2)C1 C1(NC(C2(C)N(C(CC(C=C)CC)=O)CC(O)C2)=O)CC(C)N(C)CC1C c1(C(C(C)NC(c2nc(CNC(=O)OC(C)(C)C)cs2)=O)O)cccc(Cl)c1 C1(NC(=O)CCc2ccccc2F)CC2C=CCC(C1)C2 N1(C(C(CC(=C)C)NC(c2cccc(F)c2O)=O)=O)CCn2ncnc2C1 CCC(CCC(=O)NCCN1CCCOCC1)NC(=O)CC1C=NN(C)C1=O C(CC(=O)N(C1CC(C(N)=O)C1)C)N(C(c1cc[nH]c1)=O)CC C#CC1(C(N2CCC(C(C)OC)C2)=O)CN(C(c2ccc(O)nn2)=O)C1 Cc1onc(Cl)c1C(N1CCN(CCCNC(=O)CC2(C)CC2)CC1)=O Brc1[nH]nc2ncc(-c3nc(Cc4ccccc4)nn3C3CCSC3)cc12 N1(C(CC2(COC)CC2)=O)CCCC2(C1)CN(C(c1cc(C)n(C(C)C)n1)=O)C2 N1(C(CN(C(C)C)C)=O)CC2(CCN2C(c2c(C(F)(F)F)cccc2Br)=O)C1 Cc1ccc2c(n1)CN(C(=O)CCC(CC(C)C)NC(=O)CC1C=CCC1)C2 CCC(C(=O)N1CCCC1C(C)(C)CNC(=O)Cn1nccc1C)SC C(C(=O)N=c1ccn(CCF)[nH]1)C1N(C(C=C(C)C)=O)CCOCC1 C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCN1Cc1ccc(C)cc1 N1(C(c2c(C)occ2)=O)CCN(C(=O)CC2CCC(=O)NC2=O)C(C2CC2)C1 N1(C(C2CC(C)(NC(C(C)N=[N+]=[N-])=O)C2)=O)CCC12CCC(O)CC2 N1(C(C(C)NC(CC)=O)=O)CCCC(C)(Nc2ncc(C(F)(F)F)cc2Cl)C1 N12CCCC1C(=O)NCCC2=O.C1(NC)CC(O)C1.C#CCOC c1(C(C)C(=O)NCCCCC(C)NC(C2(CF)CC2)=O)ccc(Cl)c(Cl)c1 C(=O)(C(O)C(O)C(=O)OC(C)(C)C)OCC.C123CC(CN1C2=O)C3 c1(C(C(=O)NC(C)C)N(C)Cc2scc(C)n2)ccc(CO)cc1 c1(CNC(C2C(C(=O)OC)C2)=O)cn(C2CN(CC3CC(O)C3)C2)nn1 c1(C(N2CCC(Oc3ccc(C(C)=O)cn3)CC2)=O)cccc(CC)c1F N1(C(c2c(C)c[nH]n2)=O)CC2CC(NC(C3(N4CCCC4)CCC3)=O)CC1C2 N1(C(C2CN(C(CC3CCC(C)(C)O3)=O)CC2(F)F)=O)CC2COCC2(C)C1 c1(C(=O)NCC2(F)CC(CNC(C(C)(C)CF)=O)C2)cc(N)cc(F)c1 Cc1cc2ccc(C(N3CC(C4CN(C(=O)CNS(C)(=O)=O)C4)C3)=O)cn2c1 C1(C)(C(NOCC2CC(=C)C2)=O)CC(NC(=O)CC2CC2(Cl)Cl)C1 C#CCCCCCC(=O)N(CCNC(c1cccc(C(N)=O)c1C)=O)C1CC1 N1(C(CCC(C)OC)=O)CCCC(C2CCN(C(c3c(C)cnn3C)=O)CC2)C1 Cc1[nH]c(=NCc2ccc(O)nc2)sc1C(=O)Nc1ccnc(Cl)c1Cl C#Cc1ccc(F)c(C(=O)NCC2(NC(C3(C)CCCC3(F)F)=O)CC(OC)C2)c1 CC(CN=c1[nH]c(-c2ccccc2)cs1)SC(C)Cc1ccc(Cl)cc1 C1(F)(NC(c2cc(CCC)n(C)n2)=O)CC2CC1(C(=O)NC)C2 C#Cc1ccc(NC(=O)C(C)(C)OC(C)C)cc1.N12CCC(C1)CC2=O CN1CCN(C(=O)C(=O)C2CCCC2)CC1NC(=O)C(F)(F)F.C1CCN1 C1(CNC(Cn2ccc(C)n2)=O)CN(C(=O)CC(C)(C)C2CC2)CC(C)(C)O1 C12CN(CCO1)C(=O)c1csc(c1)CNC(=O)C2.CCC(CC)n1ccnc1 Cn1ccc(C(=O)NCC2CC2CNC(=O)Cc2sc(O)nc2O)c(O)c1=O c1(C(N2CCC(NC(C(N3CCSCC3)C)=O)C2)=O)cc2c(C)sc(C)c2s1 Cc1nc(CO)oc1C(=O)NC1CCC1NC(=O)C=Cc1cscn1 C1(NC(C2(C(=O)OCC)CC2)=O)CN(C(c2ccc(C)nn2)=O)CC1C1CC1 C1(C(=O)NCCCOCCNC(CCNC(N)=O)=O)C2COCC12 C(=O)(C1CCCn2nccc21)NC1CCN(C(c2cc(CF)on2)=O)C1 c1(C(N2CC(O)(CNC(CCCOC)=O)C2)=O)cc(N)cc(C)c1F Cn1ncc2ccc(CC(N3CCCC(CC4CCCNC4)C3)=O)cc12 CCCCCCCCNC(=O)CC(CNC(C1CCC(C)(C)OC1)=O)C1CCC1 n1(CC(=O)N(C(C)CNC(C2CCN2C)=O)C)ccc(O)nc1=O c1(CC)ccc(C=CC(=O)NCCN(C(=O)CSc2nccn2C)CC2CC2)o1 c1(CNC(C(C=C)O)=O)cccc(C(=O)N(C)CC2CCCOC2)n1 Cc1cccc(C)c1CC(N1CCC(CF)(NC(=O)C(F)=CCCF)C1)=O n1(CC(=O)NC(CN(C(=O)CCC2(C)CC2)C)C2CC2)ccccc1=O CCCC(CC)CCC(=O)NCC1CCN1C(c1ccsc1)=O n1(CCCC)cc(C(c2nnnn2C2CC2)N(C(C)(C)COC(C)C)CC)nn1 C(CN=c1ccc(C(=O)NCC2CN(C(C3CCCC3OC)=O)C2)c[nH]1)OC C1(NC(c2c(C)nncc2)=O)CCC2(CC1)CC(NC(=O)CCn1cccc1)C2 C1(CC2CCC2)C(=O)N1C.n1(CC)cc(C2(C)CCCC2)nn1 C12(NC(c3ccnc(F)c3F)=O)CCCCCC1N(C(=O)Cn1ccnn1)CC2 C1(NC(=O)CNC)CC2(C1)CC(C(N1CCC(=C)CC1)=O)C2 C(=O)(CCS(N)(=O)=O)N1C(CC)C(C(=O)NCC2CSCCO2)CC1 C12(CNC(c3c(CCC)n(C)nn3)=O)CN(C(C3(CC)CCC3)=O)CC1CCO2 C1(NC(C2N(C(=O)C=Cc3ccncc3)CCN(C)C2)=O)CCn2nccc2C1 Cn1c(O)nc2ccc(C(=O)NC(CNC(C3CC34CC(O)C4)=O)CO)cc12 C1(C(=O)NCC2(C)N(C(CCn3c(C)cc(C)n3)=O)CCC2)CC(C)CC(C)C1 Cc1ccc(C(=O)NC2CC(F)(CNC(=O)C(C)(C)CO)C2)cc1N1CCCC1 C1(C(N2CC(O)(CN(C)C(c3ccc(F)c(F)c3)=O)C2)=O)C(F)(F)C12CCC2 C(=O)(C(F)(F)C(F)(F)F)N1CC(CN(C(=O)C=Cc2cc(F)cc(F)c2)C)C1 c1(C(N2C(CNC(C3(CCC)CCC3)=O)CCC2)=O)ccc(Cl)cc1O CN=c1[nH]cc(C(=O)NCCN(C(=O)Cc2cccc(SC)c2)C)s1 CCCCC(O)C(=O)Nc1ncc(-c2ccc(N)c(NC(=O)CC#N)c2)s1 c1(C(=O)NCC(C)N(C(C(C(C)C)c2ccc(F)cc2)=O)C)cccc(=O)n1O c1(C(=O)NCC2C(NC(CCc3ccc(C)s3)=O)C2)ccc2oc(C)nc2c1 c1(C(=O)NC2(CCC=C)CCCC2)ccc(S(=O)(=O)N2CCOCC2)nn1 C1(C(=O)NC2C(C)(CN(C(CCCC=C)=O)C)CCC2)CN2CCN1C(C)C2 C1(CNC(C(CCOC)NC(C(CO)OC)=O)=O)CCC=CCCC1 C1(C)(C(N2CC3(CN(C(C(C)OC4CCOC4)=O)C3)C2)=O)CCCCCCC1 c1(C(=O)NC(C2CCCN2C(C2CNC(=O)N2)=O)C)coc(-c2ccccc2)n1 c1(C(N(CC(C)(C)NC(c2ccc(N)c(N)n2)=O)C)=O)c[nH]nc1S(N)(=O)=O N1(C(Cc2cn(CC)nc2)=O)CC2(CC2)CC1CNC(C1(CCOC)CCC1)=O C(=O)(CS(=O)(=O)CCO)NCC1C2CN(C(c3ccn(C)c3)=O)CC21 CC(C(=O)NC(C1CCN(C(C2(C#N)CCCCC2)=O)CC1)(C)C)C1=CCCC1 C=CCCC(C)(C)C(=O)NCc1cn(CC(=O)Nc2ccc(NC(C)=O)cc2)nn1 CCC(CC(F)F)C(=O)NC1CCN(C(=O)CCSCC(N)=O)C1 C(=O)(CCCCCC(=O)OC(C1COCCO1)=O)NCCCNC(=O)OC C1(CCNC(c2ccnc(CNC(C3CCC4(CC4)C3)=O)c2)=O)CCCC2CC12 c1(CC)ccc(C(=O)NC2(C(=O)NCCC(=O)NO)CC2(C)C)cn1 c1(OC)ccc(CNC(c2nc(-c3ccc(Cl)cc3)no2)C)c(F)c1 N1(C(CCNC(COC)=O)=O)CCCCC(N(C(=O)C(C)(C)CO)C)C1 C(=O)(C1CCOc2ccc(Br)cc21)NC1(CO)CN(C(CCC#C)=O)C1 Cc1cnc(C(=O)NCC2CCCC(NC(c3[nH]c(C)nc3C)=O)C2)cn1 c1(OCC#C)ccc(C(N2CCOC(CSC)C2)C(=O)NC(C)C)cc1OC N1(C(c2cc(CC)no2)=O)CCCC(C)C1CNC(=O)CCc1cnn[nH]1 c1(NC2CC(O)(CNC(c3ccc(C)nn3)=O)C2)cc2nnc(C)n2cn1 C(=O)(CC(C)CC(=O)NCC1(C)CCCN1C(C1CC2(CCCC2)CO1)=O)OC c1(CN(C(C2Cc3nccn3C2)=O)CC)cc2cc(OC)c(OC)cc2[nH]1 c1(C(=O)NC(C2CCN(C(c3cn[nH]c3)=O)CC2)C)c[nH]c2nccc-2c1 c1(C(N(C2CCCN(C(=O)CC(C)(C)O)C2)CC)=O)n[nH]c2ccccc12 c1(OC)ccc(C(N(CCO)CCn2cnc(=N)[nH]2)=O)c(Br)n1.C(CCC1ONC1)N C1(COC)CC(CNC(c2ccncc2)=O)N(C(c2cnc(C(C)C)nc2)=O)C1 C12(NC(CCc3ccc(C)o3)=O)CC1CN(C(=O)CC1CCOC1=O)C2 c1(CC(C(=O)NC(C)CNC(=O)CC2(O)CCC2)F)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(C)CCC2CCCC2)cccnc1CNC(=O)C(C)(C)C C(CC(C)C)(C(=O)N1CC2CC1CN2C(C)C)NC(Cc1scc(C)c1)=O C1(C(=O)NCC(=O)NCCOC)CC(C)CN(C(C2(CO)CCC2)=O)C1 c1(CC(=O)N(CCCNC(c2ccc(C)cc2O)=O)CC)nn(C)cc1[N+](=O)[O-] N1(C(C)=O)CCN(C(=O)CC2(NC(=O)C(F)F)CCC2)C(C)C1 C(=O)(C1=CC2(CCOCC2)C1)NC1C(CNC(c2cn(CC)nc2)=O)CCCC1 c1(C(=O)NCC2C(NC(CN(C3CCCC3)C)=O)CC2)ccn(C)c(=O)c1 c1(C(=O)NCC2C(CNC(C=CS(C)=O)=O)C2)nnc2ccccc2n1 C1(NC(c2c(CNC(c3ccnc(CO)c3)=O)noc2)=O)CCC2CCCC1O2 C=CCC(C(=O)N(CC(=O)NOCCN(C)C)CC1CCCC1)OC Cc1ccc(C)c(C(=O)NCC2CC(NC(C3(C)CCCS3)=O)C2)c1N C(=O)(C(C)(C)C(C)NC(=O)C(C)=C1CC1)NCC(=C)C c1(C(=O)NC2C(NC(c3ncn(C(C)(C)C)c3)=O)CCC2)ccc(Cl)c(Cl)c1O Cc1sc2c(F)cccc2c1S(=O)(=O)NC1CCCC(O)C1O C(CC(C)(C)C)(C(=O)N(CCC(=O)NC(C1(O)CCCCC1)C)C)NC(C)=O Cc1ccc(N(CCN(C)CCO)NC(=O)Cn2cc(C(F)(F)F)cn2)s1 C1(OC)CC(C(=O)NCc2ccc(O)cc2)N(C(c2ccc(F)cc2)=O)C1 c1(C(=O)NCC(COCC)(O)CO)cccc2cncn12 c1(OCC(=O)NCCCC(C)(C)NC(CC(C)(C)O)=O)cc(F)cc(F)c1 C(CCC(=O)NCC(C(C)C)NC(=O)CN(c1ccccc1)CCOC)=CC c1(NC(C2(C)CCN(C(CCSCC)=O)C2)=O)cc(C)cnc1C C1(CNC(C2(F)C3CCCC23)=O)CCCCN(C(C2CN3CCC2CC3)=O)C1 CC(C)CCCC(=O)NC(C1CCCC1)CNC(=O)C(CC(F)F)C1CCC1 c1(NC)cnc(C(=O)NCC2CC(CNC(C3CCC(C)C3)=O)C2)cn1 CON(CCC(=O)NCC(C)N(C)C)C(=O)C1(Cl)CC1(F)F N1(C(CC2C(C)CCCC2)=O)CCC2(NC(C3CCCC(=O)N3)=O)CCCC12 c1(C(=O)NCC2C(C(=O)NCc3nc(C(C)C)on3)CCC2)ccc(C#N)s1 C1(CN(C(C(C)OCCOC)=O)C)CCCN(C(c2nocc2C(C)(C)C)=O)C1 C(=O)(CCCC(=O)c1ccccc1N)N(c1ccccn1)CC(=O)O.c1(S)ccccc1 C(C(=O)NC1CC1)(C1=NOCC1)N1C(C)CCC(C(=O)OC)C1 N1(C(=O)NCCC2(NC(COC)=O)CC2)CCCC2CN(C(C)=O)CC12 N1(C(c2[nH]c(=NCC)sc2)=O)CCCN(C(=O)C(CC)C2CCC(=O)N2)C(C)C1 N(C1CSc2ccc(Br)cc21)C(c1c[nH]c2c(Br)cccc12)=O Cc1cc(N2CC(CO)OC(C)(C)C2)nc(=NC(C)CC(C)(C)C)[nH]1 c1(C(=O)NCCCCCNC(C(C)(C)OCC)=O)cc(N)c(C)c([N+](=O)[O-])c1 C1(NC(CC=C(C)C)=O)C=CCC(C(=O)NCC2(F)CCOCC2)C1 N1(C(c2c(C)nns2)=O)CCC(C)C(CC(=O)N(C2CC(O)C2)C)C1 N1(C(COCCOCCOC)=O)CCC(O)(CCNC(c2cc(F)c[nH]2)=O)C1 C1(C(=O)NC(CC=C)CC)CN(C(=O)CCC(C)N(C)C)CC1(C)C c1(OC)cc(C(=O)NCCNC(=O)C#CC(C)(C)C(C)(C)C)c([N+](=O)[O-])cc1OC c1(C(=O)NC2CN(c3nccc(SC)n3)CC2F)ccc([N+](=O)[O-])nc1 N1(C(C(c2cccnc2)C)=O)C2CCC1C(CNC(=O)CC1CC1)C2 C12(OC)CCC(C(N3CCC(N)CC3)=O)(CC1)C2.C(=O)(CCOC)N(CO)CC1CC1 CC1(C(=O)N(CC(CC2CC2)C(=O)O)c2cnn(CC(F)F)c2)CCCN1 c1(CN(C(c2c(C)nccn2)C)C)ccc(F)c([N+](=O)[O-])c1 c1(C(N2CC(NC(=O)Cc3nonc3C)CC(OC)C2)=O)cc(N)c(F)cc1F C12(C(=O)NC3C4CN(C(COCCC)=O)C(C4)CC3)CCC(N(C)C)(CC1)CC2 CCC(C(=O)NC1CN(C(C2(CSc3ccc(F)o3)CC2)=O)C1)OC1CCCC1 C#Cc1ccc(C#N)c(NC(=O)NC(c2cnnn2C)CC)c1 CN=c1nc(N2CCC(Oc3cccnc3)C2)[nH]c(=NC2CCCSCC2)[nH]1 C1(N(C(C2(CCCF)CC2)=O)C)CCCC1C#N.C1(C(=O)NCC)CC(CF)C1 c1(C(=O)NC2(C)CN(C(C3CCC(OC)C3)=O)C2)noc(C)c1C c1(OC)cnccc1C(=O)NCC(N1CCC(C2CCCCO2)C1)=O C(CC(C)C(=O)NCC(F)CNC(C1CCN(CC2CC2)CC1)=O)=CCC C12CN(CC3(CCC3)C1)C(=O)N2.c1(CC)cc(=NCC2CC(=O)NC2=O)[nH]cn1 C(CCCCC(=O)NC(=O)CCN(C)CCO)NC(CC)Cn1cncn1 Cc1ccc(NCC(=O)NC(C)CC(C)NC(c2cnn(C)c2)=O)c(C)c1 CC(O)C(C)(C)C(=O)N1CC=CC(NC(=O)CCC2CCCCO2)C1 Cc1c(C(=O)NN2CCCOCC2)cnn1CCc1cn(CCCC(=O)O)nn1 C1(CC(=O)NCc2ncn(CC)n2)CC(NC(=O)C(C)C)C1(C)C CS(=O)(=O)c1cc(C(=O)NC2CC3CCC(C2)N3C(c2cc(F)n[nH]2)=O)co1 C=C=CC(C)C(=O)NC1(C(=O)NCC23CC(F)(C2)C3)CC1(C)C c1(NC(C(=O)NCc2onc(COC)n2)=O)ccc(C(C)(C)O)c(F)c1 c1(C(N2CCC(C)(NC(C3CNC(=O)C3)=O)C2)=O)cc(Br)cc2c1CCN2 c1(N(CC(C)(C)OC)C)nc(NCc2cncn2C)c2c(n1)c(C)nn2C C(N=c1[nH]c(C(=O)OC)c(CC)s1)C12OCC(NC(c3n(CC)cc(Cl)c3)=O)(C1)C2 N1(C(COCC(=O)OC)=O)CC2CCC(CNC(C3COCCOC3)=O)C2C1 N1(C(CNC(=O)CN2CCOCC2)C(F)F)CCN(C(c2ccccc2)=O)CC1 C1(C(C)NC(C2(C(N)=O)CCC2)=O)CN(C(=O)C=Cc2ccsc2Br)CCO1 C1(CC)CCCCC1C(=O)N(CCCOCCN(C)C(c1ccncc1Cl)=O)C c1(CNC(C(COC)O)=O)ccc(CNC(c2ccc(CO)c(C)c2)=O)c(F)c1 Cc1coc(C(N2CCCC2C(C)(C)C(=O)NC2CCC(N(C)C)C2)=O)c1 N1(C(c2nc(C)oc2)=O)CC23CCCCC2(C1)CN(C(C1(C#N)CC(=O)C1)=O)C3 C(CCCCCNC(=O)CCOC1CC1)N(C)C(C1CC2C=CC1C2)=O C(=O)(CCC(C)(C)OC)N1CCC(C(C)NC(c2c(OC)nsc2)=O)C1 C1(C(=O)NC(C)C(O)C(C)C)(CNC(C(CO)OC)=O)CC2(CC2)C1 c1(NC(C2C(C(F)(F)F)C3CCC2O3)=O)cnc2n[nH]c(Br)c2c1 c1(OC)nccc(C(=O)NCc2cc(C(=O)NC(C)C(C)n3cncn3)n(C)n2)n1 c1(COC)cc(NC(=O)Cc2ccc(N)cc2)n(-c2ccccc2)n1 c12ccc(cc1)OC2.C(CCCCNC(C1CC1F)=O)N(C)C(c1ccoc1)=O N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3(C)CC(C)=NO3)=O)CC2)C1 Cc1cc(OCCC(N2CCCC(NC(=O)C#CC(=O)O)C2)=O)cc(C)c1 Cc1ccc(C(N2CCCCCC2CNC(=O)C(F)CC2CC2)=O)cc1F CCC(C)C(O)C(=O)NCC1(O)CN(C(c2ccc(-c3ccnn3C)cc2)=O)C1 N1(C(c2c(C)nccn2)=O)CC2(CCC2NC(C2CC23CCCCC3)=O)C1 C1(C(=O)Nc2c(C)cc(CO)nc2)CCC(C)(C)N(C(=O)CC(=O)N(C)C)C1 C1(CNC(C2CC(C#C)(O)C2)=O)(NC(=O)C(C)N(C)CC)CC2CCC1CC2 C(=O)(C1CCc2nccn21)NCC1(O)CCCN(C(CNC(N)=O)=O)CC1 C1(C(=O)NCCOC2CCN(C(=O)CC(F)F)CC2)CCn2nncc2C1 C(=O)(C1CCCn2c(C)cnc21)NC(CNC(c1cccc(SCCC)c1)=O)C C1(N(C)C(=O)OC(C)(C)C)CCS(=O)(=NC(=O)c2ccsc2)C1 c1(Cn2cc(C3(O)CN(C(=O)CC4CC5CC5C4)C3)nn2)cnc2sccn12 c1(OC)cc(C(N2CCC(C)(NC(=O)COCC3CC3)CC2)=O)cc(F)c1 Cc1c(Cl)cnn1CC(=O)NCC1CCCC1NC(c1ccccc1C(F)F)=O C1(CNC(CC(C)OC)=O)CC2CCC(C1)N2C(C12CCC(C1)C2)=O c1(C(=O)NCC(C)(C2CC2)NC(c2n(C)c(Cl)c(Cl)c2)=O)c(F)ccc(Cl)c1N C1(C)(CC(=O)NC2CC(N(C(=O)CCC3CCCC3)C)C2)CCOCC1 CCC(C)(CCC(C)C)C(=O)N1CC(C2(NC(=O)COc3ccon3)CC2)C1 n1(CC(C)C)nc(C2CC2)nc1-c1cc(Br)cn1C(F)(F)F CS(=O)(=O)C(CNC(c1ccc(C#N)cn1)=O)CNC(C12CCCN1CCC2)=O c1(C(C)C(=O)N2CC(C(C)NC(C3(C)CC3Br)=O)C2)ccccc1F c1(OC)cc(N(C)CC2CCCN2C(C2CC2(C)C(C)C)=O)nc(OC)n1 C(=O)(C(F)C(F)(F)F)NCCN(C(C1CCCC1C1CC1)=O)CC Cc1ccc(C(N2CCOC(Cn3cc(CO)nn3)C2)=O)c2ncccc12 c1(C(=O)NCCCN(C(C2(F)C(C)C2)=O)C)c(Br)c(C2CC2)nn1C(C)C C1(CCNC(C2C(=C)C2)=O)CN(C(c2sc(C)nc2Br)=O)CCO1 C(=O)(C(C)(C)CCCN=[N+]=[N-])NCC(C)NC(COCc1ccc(C)cc1)=O c1(N(CC(C(=O)OCC)C)C)nc2cc[nH]c2c(=NCCNC(=O)CCN)[nH]1.NC C(=O)(C#CC1(C)CCCO1)N1CC(O)(CNC(CN(C)C(c2cccs2)=O)=O)C1 Cn1cc(C(=O)NC2CN(C(=O)CC3CCOC3)C(C)(C)C2)c2cc(F)ccc12 C1(C)(C(=O)NCCS(=O)(=O)NCC)CN(c2cnn(C)c2)C1=O c1(C(CC)C(=O)NCc2nccc(N3CCOC(CN)C3)n2)ccc(F)c(F)c1 C(=O)(C1=NOC(C)C1C)N(CC(C)NC(c1c(OC)ccnc1O)=O)C Cc1csc2c(C(N3CC(CNC(C4CC4(C)C)=O)C4(CC4)C3)=O)cccc12 CCC(COC)C(=O)NC(CC1CC1)CC(=O)N(C(C)COC)C N1(C(C23C(C(N)=O)(CCC2)C3)=O)CCC2(CC1)CC2NCC1CC12CCOCC2 CC1CC(NC(C2CCOC2=O)=O)CCN1C(c1ccc(CN=[N+]=[N-])cc1)=O N1(C(CC(C)(C)O)=O)CCN(C(=O)C=CC2CCCCC2)CC1C1CCCC1 C12(C(N3CC(=CCC)C3)=O)CC(CCO1)N(C(C1CCCC(=O)N1)=O)C2 N1(C(c2cc(CCC)[nH]n2)=O)CCC2CCN(C(=O)CSC(F)F)C2C1 C(=O)(C(C)C(C)(C)C)NCC1(O)CCN(C(c2c(SC)snn2)=O)C1 C1(NCC(F)(F)F)CCCCN1C(C(C)N(CCCC)CCOC)=O c1(NC(=O)NCC(C(C)O)C)cccc(-c2csc(N3CCOCC3)n2)c1 C1(C(N2CC(C(C)NC(=O)CCCCCF)OCC2)=O)CC2CC2CC1C C#CC1(C(=O)N(C)CCC#CC)CCN(C(=O)CCOCC(C)C)CC1 C(CCNC(=O)C(C)N(C)C)(C(=O)NC(c1nc(C)cs1)C)OC CC1CCN(C(c2ccc(C(F)(F)F)nc2)=O)C1CNC(C1CC=CC1)=O C1(C(N2CCCC(F)(CNC(c3ncc[nH]c3=O)=O)C2)=O)CCOC2(CCC2)C1 C1(NC(c2c(SC)nn(C)c2)=O)CCN(C(=O)CC2(C)CCC2)CC1F C12(C(=O)NC3CN(C(Cn4c(C)ncc4)=O)CC3C)CCC(N(C)C)(CC1)CC2 C(=O)(C(C)C(C)C)OCC.C12(CC(=O)C1)C(=O)N2.C(=O)(CC(=O)O)N.C1(=O)NCCN1 C(=O)(C(C)C1=CCCC1)NC1(C)CCN(C(c2c(N)ccc(C)c2)=O)C1 CC1=C(C(=O)NC2C3CCN(C(=O)CC4CCOC(C)(C)C4)C23)CCC1 c1(C(C(=O)N(CCC)CCNC(C23COCC2C3)=O)C2CCCC2)ccccc1 C1(CNC(c2ccc([N+](=O)[O-])s2)=O)CN2CCCCC2CN1C(c1cscn1)=O N1(C(=O)OC(C)(C)C)CC(CC2(CO)CC(=O)N(O)C2)OC2(CCC2)C1 N1(C(CSC)=O)CC2(CCOCC2)CC1CNC(C1CC1(C)CC)=O CCC1=NOC(C(=O)N(C2CCCN(C(=O)C3=CSCS3)C2)C)C1 N1(C(c2n(CC)ccn2)=O)CCC2CCC(C1)N2C(c1coc(C#N)c1)=O CC1CN(C(=O)C(C2CCCCC2)C)CC1C(=O)NCCc1cnn(C)c1 N1(C(C2(OC)CCCC2)=O)CC(C(=O)NCCc2ccn(C)n2)C(C2CC2)C1 O=C(CC1=CCCCC1)NC1(c2ccon2)COC1 C12(C(=O)NCCN(C(=O)Cn3nnc(=N)[nH]3)CCOC)CC1COC2(C)C C1(C(=O)NCCCNC(CO)=O)(N)CC2CCC1C2.C=CCCC(=O)OC(C)(C)C C1(NC(Cc2ccc(C)s2)=O)COC2(C1)CN(C(=O)CCCc1n[nH]c(=N)s1)C2 CC(F)(F)CCC(=O)NC1CCC(NC(C2CCOC2c2ccnn2C)=O)CC1 C(=O)(C1CCCc2cncn21)NCCCCNC(c1cc(C)c(F)cc1F)=O C(=O)(C1Cc2cccc(Cl)c21)N(C(CNC(Cc1ccn(CC)n1)=O)C)C N1(C(C(CCC)NC(C)=O)=O)CCc2c(c(COC)nn2C)C1 c1(C(=O)NC2(C)CN(C(C3CNC(=O)C3)=O)C2)cnc(S(C)(=O)=O)s1 CC(C)(C)CC(O)CC(=O)N1CCCC(C)(NC(=O)CCOCC(F)(F)F)C1 Cc1cc(C)c(C(N2CCNC(C(N3CCC(Cl)C3)=O)C2)=O)c(Cl)n1 Cc1cc(C(=O)N(CC(C)(C)CNC(C2CC(N3CCCC3)C2)=O)C)ncc1N C1(CC(N2C(C(=O)NC)CC2)=O)CCN(C(c2ccnc(C(F)F)c2)=O)CC1 C1(CNC(CC(=O)N(C)C)=O)CN(C(C2(C)CCN(C)C2=O)=O)CC2(CCC2)O1 N1(C(Cc2c(C)non2)=O)CCCC2CN(C(=O)CC3CSCCO3)CCC12 CC(C)C(O)C(C)(C)C(=O)N1CCC(NC(C2CCC(N(C)C)CC2)=O)C(O)C1 c1(CC)c(Nc2cccc(OC)c2OC)cccc1C(=O)N(C1CC1)OC CC(C)C(C)(CNC(c1cc(CO)on1)=O)NC(=O)CSc1nnc(S)n1C C(=O)(NN1Cc2ccc(Br)cc2C1=O)c1ccc(C#C)cc1OC c1(CN=C(NC(CC)C)NC2CCCC2(F)F)ccc(F)cc1O CC(CC1CCCO1)N=c1[nH]c(=NC(C)Cn2ccnc2)c2cc(Cl)ccc2[nH]1 C(=O)(CCCCCCC)NC(CCCC)C(=O)NCc1ccsc1 C1(CC)CC(c2ccccc2)CN(C(c2cnn(C3CCCN3)c2)=O)C1 C(CCN(C)C(C1CC1c1ccccc1F)=O)(C(C)C)NC(C(COC)C)=O c1(CN(CCOC)CCNC(=O)COC)cc2cc(C)ccc2nc1Cl C1(C(=O)NC2CCC(CNC(c3ccnc(CO)c3)=O)CC2)SC2C=CC1CC2 CC1C(NC(=O)C(C)S(C)(=O)=O)C(C)CCN1C(C1CN(CC(F)(F)F)C1)=O C(=O)(CCCCCNC(=O)C(c1ccccc1)C)NCc1n(CC)ncn1 CC(C)(C)C(O)C(=O)NC1COCC1CNC(c1cnn(C2CCC2)c1)=O N1(C(C=CC(=O)N(C)C)=O)CC2(C1)CN(C(=O)CCc1cnco1)CC2CO Cn1c(NC(=O)Nc2cccc(C3CC3(F)F)c2)nc2cccc(F)c12 N1(C(C(C=C)O)=O)CCN(C(c2nccnc2C(N)=O)=O)CC1c1cn[nH]c1 c1(C(N2CC(C)C(NC(c3cccc(F)n3)=O)C2)=O)c(F)cncc1Cl C1(N(C(=O)NCc2ncc(CC)s2)CC2CCOCC2)CCS(=O)(=O)C1 C(CCCCCCCO)=CC(=O)NCC(C(C)C)(C)NC(=O)CCOC1CCC1 c1(OCC)ccnc(NCCC2CCCCN2C(c2cc(CO)oc2C)=O)n1 C(C)(CN=c1[nH]c(C)cc(=NCC2CC3CCCC(C2)C3)[nH]1)OCCOCC N1(C(Cc2ncc(CC)[nH]2)=O)CCC(O)(CN(C(=O)CCC(C)C)C)C1 C1(NC(C2C(NC(=O)OC(C)(C)C)CC2O)=O)CC2CCC(C1)N2 C1(CC(=O)N(CC(CC)NC(=O)Cc2ccnn2C)CC)CC(C)(C)CO1 Cc1cccc(C)c1S(=O)(=O)NC1(C(=O)N=c2cc[nH]cc2)CCC1 N1(C(c2ccc(CSCC(C)C)o2)=O)CCCCCC(NC(=O)CNC=O)C1 c1(N)cnc(O)c(Br)c1.CC1(CC(=O)NCCNC(C2(C)CC2)=O)CCCCC1 Cn1cc(NC(=O)CC2CC(NC(c3cccc(Cl)c3)=O)C2(C)C)c(C#N)n1 C(=O)(C1=NOC(C)(C)C1)N1CC(C(C)C)N(C(C2(C(F)(F)F)CC2)=O)CC1 Cn1c(C(N2CC3CC3(NC(c3cccc(C(F)F)c3)=O)C2)=O)cnc1[N+](=O)[O-] c1(CC)cccnc1C(N1CCC(C(C)C(=O)NC(C)(COC)C2CC2)CC1)=O C(=O)(C1(C)CCn2ccnc21)N(CCn1cc(Cn2ccnn2)nn1)CC.C1CC1 c1(C(=O)NCC(CNC(CCCCC)=O)OC)ccc2cnc(C)cc2c1 C1(CC(=O)NC(c2ccc(CNC(c3cc[nH]n3)=O)cc2)C)COC(C)(C)CO1 c1(C(=O)NCC(C)N(C)C(C23CC2COC3(C)C)=O)ccc(C2CC2)c(F)c1 N1(C(c2cnn(-c3ccccc3)c2N)=O)CCN(C(C)=O)C(C)C1.C1(OC)CO1 N1(C(Cc2c(C)ocn2)=O)CC2CCC(C1)N2C(=O)CCN1CCCS1(=O)=O c1(NCN)ccc(C)nn1.C(C(=O)NC1COC1)(C1CCCC1)OCC.CC C1(C(=O)NC(CC=CC)C(=O)N2CCCC2CNC(N)=O)CCOCC1(C)C N1(c2cc(C)nc(C3CC3)n2)CC2(C1)SCCC2NC(=O)CCC(C)N(C)C Cc1ccc2cc(C(N3CCCN(C(=O)C(C)C)C(C)C3)=O)cnc2c1 N1(C(CC(=O)NCC#C)=O)C2CCCC1CN(C(c1cc(F)ccc1F)=O)CC2 c1(C(=O)NC2CCN(C(C(CC)Oc3ccccc3)=O)C2)ccc(CO)c(F)c1 C1(CNC(C2(CC(C)C)CCC2)=O)C2CN(C(=O)C(C)(C)C3CC3)CC12 c1(NCC2CCC(NC(CCC3C(=O)NCC3)=O)C2)ncc([N+](=O)[O-])cc1Br c1(C(=O)NCC(C)CNC(=O)C=CC2CCCO2)cc(N)c(F)cc1Cl N1(C(C2(C3CCCO3)CCC2)=O)CCCC1C(=O)NCC.C12COCC1CN2 CCN=C(NC1C2CN(C(C)=O)CC12)N1CCC(C)(F)C1.C1(C2CN2)CCCC1 C(=O)(C(F)(F)C(O)c1ccc(F)cc1)NCC1N(C(=O)CCF)CC(O)C1 CN1CCOC(C(N2CC(O)(CNC(C3CCN(C4CC4)S3(=O)=O)=O)C2)=O)C1=O N1(S(c2ccc(OCCC)c(CC)c2)(=O)=O)CCc2c(ccnc2Cl)C1 c1(CC)cc(C(N2CC(CNC(C3SCCS3)=O)(COC)C2)=O)ns1 n1(CC)nc(C(C)C)cc1C(=O)NC1CCN(C2CNC2)C1=O CCC(C)(C(=O)NC(C)C(C)(C)NC(=O)CCc1cc(Cl)cc(Cl)c1)C(N)=O C1(CC(=O)N(C(CO)CO)C)CCCN(C(=O)C(c2ccccc2)O)CC1 C1(OC)CN(C(=O)OC(C)(C)C)CC1C(=O)OC(C(F)F)OC N1(C(C(CCC)NC(N)=O)=O)CC2CC(C1)N(C(c1cc(C)nc(Cl)c1)=O)C2 N1(C(COc2cc(C#C)oc2)=O)CCOCC(C)(C)C1 CCC(C)CCCCC(=O)N1CC2(CCC2)CC1C(N1CCC2(CC(=O)NC2)C1)=O CCC(O)C(C)C(=O)N1CCC(CCNc2cc(C(C)C)nc(C)n2)CC1 c1(CN2CC3N(C(c4cc(C(C)C)no4)=O)C3C2)cc(O)c(O)c(O)c1 N1(C(C2CCN(C(C(CCC)OCC)=O)C2)=O)CCN2CC(O)CC2C1 C(CC(C)C(=O)N1CCCCC1CNC(c1sc(N(C)C)nc1C)=O)=CC CCC(CNC(=O)COC1CCN(C(=O)CCCCNC(N)=O)C1)CC(C)C CCCCCCC(C)CC(=O)N(C)CC1(O)CN(C(=O)C(C(C)C)OC)C1 C(CN=C(NCC1CCCOC1)NCc1nnnn1-c1ccccc1)OCC C(=O)(C(C)(C)C(c1nnnn1C1CCCCC1)NCC1CCS(=O)(=O)CC1)OC c1(OC)cc(C)c2cc(C(=O)NCC(O)CNC(=O)CN3CCCCC3)oc2c1 C1(N(C2CCC(CO)CC2)C(C)=O)CC2CCC1(C(N1CCC(C#N)C1)=O)C2 N1(C(C(CC=CC)C)=O)CCCC(C(=O)NCC(CC(C)C)N(C)C)CC1 c1(OC)c(C(=O)NC(C)CC2CCN(C(=O)CC(C)C)CC2)cccc1C CC(C)C(C#N)C(=O)NC(Cc1cnn(C)c1O)C(N1CCOCC(O)C1)=O CC1OCCN(C2CC3CC2CC3(O)C(F)(F)F)C1(C)C N1(C(C2ON=C(C)C2c2ccccc2)=O)CCCC(NC(=O)CC(F)F)CC1 C(=O)N(C(C1(COC)CC1)=O)C.C(C)(C(C1CC1)OC)NC(C=C)=O n1(CC)c(C(=O)NCCC2CCCN(C(c3ccncc3Cl)=O)C2)cnc1O c1(C(=O)NC2(c3ccccc3)CCN(C(=O)C3CC3)C2)ccc2c(c1)CCOC2 N1(C(c2cc(OC)c(O)cc2)=O)CCC2(CC1)CCN2Cc1cnc(Cl)cc1F c1(C2N(CC3(NCC)CCC3)CC2)nncn1C CCCCC(C)C(=O)NC1CC(O)(CNC(C2(C)CS(=O)(=O)C2)=O)C1 N1(c2ccnc(NC(c3ccc(OC)cc3)C(C)C)n2)CCCC(C)(OC)C1 N1(C(CCCC)=O)CC2CCCC1(CNC(C1CC(C(=O)NC)C1)=O)C2 N1(C(C2CC(C(=O)OC)C2)=O)CC2(CCCC2NC(=O)C(C)SC)C1 O=C(N1OC2CCC1C(O)C2O)c1ccc(N2CCOCC2)cn1 CC(C)CC(S(=O)(=O)NNC(=O)c1cn(CC(=O)N(C)C)nn1)c1ccccc1 CC(C)C(C(=O)N1CC(NC(=O)CN2CCCC2=O)C1)NC(=O)CC12CCCC1C2 C12(C(N(C(CNC(C(c3c(C)cccc3)C)=O)C)C)=O)COC(CCO1)C2 CC1CC(NC(=O)C(C)(C)CN(C)C)CN1C(=O)CC(C)(C)c1ccc(F)cc1 C(C)(C)(CCCCNC(=O)C(F)n1ccnc1)NC(c1nc(C(C)C)sc1)=O C1(C(=O)NC2(CNC(CCC(C)N(C)C)=O)CC2)CCCCCS1(=O)=O C1(F)(CNC(C(=Cc2cn[nH]c2)C)=O)CCCN(C(=O)C(O)C(F)(F)F)CC1 N1(C(c2c(C)c[nH]c2)=O)CCC(C(C)NC(c2c[nH]c(C(F)(F)F)c2)=O)CC1 C(c1cnn(C)c1C)=CC(=O)NCC1C(NC(C2(COC)C=CC(CC)=C2)=O)C1 c1(C(C(=O)NC)NC(CN(CC)CC)C)cccc(OC)c1Cl C(=O)(C(CNC(=O)C(F)C(C)(C)O)C(C)C)NCC1(CCC=C)CC1 C1(C(=O)NC2CCCN(C(CCc3n(C)cnn3)=O)C2)CC2(CCCC2)CO1 N1(C(=O)NCc2ccc(C(=O)OC)nc2)CCN(C(=O)C(C)O)CC(C)(F)C1 C(CCC(C)(C)C(=O)NCCc1nc(C)no1)NC(c1ncn(CC)n1)=O c1(CNC(COCC(=C)C)=O)cc(O)nc(CNC(=O)C(C)C(C)C)n1 c1(CCC)nc(-c2cc(-n3cccc3)c(C)o2)n(Cc2ccc(COC)cc2)n1 c1(NC(N(CCC(=O)N(C)C)CC=C)=O)cncc2[nH]ccc12 C#CC1(NC(=O)CC2CC(C)N(C(=O)Cn3ccnc3)C2)CCC(C)CC1 C1(CNC(=O)C=Cc2nccs2)CC(O)CN1C(=O)C1=CCCS1 C1(N(C2CN(C(=O)CC(c3ccc(F)cc3)C)C2)C)CCc2nnnn2CC1 c1(C(=O)NCCC2(NC(C(COC)C)=O)CCC2)c(Br)cnn1C c1(C(N2CCC(CN(C)C(C3CC3(Cl)Cl)=O)C2)=O)ncncc1N Cc1cc(F)ncc1C(=O)N(CC(C)CNC(=O)CSCCC(F)(F)F)C C1(CC(=O)N(C2C(C)CC2)C)N(C(c2cc(C(N)=O)c[nH]2)=O)CCC1(C)C c1(CNC(C(N2CCCC(CCC=C)C2)=O)=O)c(C)sc(C)c1C CC12C3C4C1C1C2C3C41C(=O)NC1CCC(NC(c2cc[nH]c2)=O)C1 N1(C(CNC(=O)OC)=O)CC(F)CC1CNC(=O)CCC1CCCOC1 C1(O)(CNC(C(CNC(CC(C)(F)F)=O)CC2CC2)=O)CCCC1(C)C C1(NC(CCC2CCN(C(C3C(C)C(=O)C3)=O)C2)=O)CC(=O)N(C)C1=O Cc1sc(S(N)(=O)=O)cc1C(=O)NC1CCCCC1NC(c1cccc(N)c1)=O C(=O)(C1=CCN(C(c2cc3ccccn3c2)=O)CC1)N(C1CSC1)C N1(C(Cc2cccc(SC)c2)=O)CC2(CC2)CC1C(=O)Nc1ccsc1 Cc1cc(=NCc2ccnn2C(F)(F)F)[nH]c(=NC2CCC3(CCC3)CC2)[nH]1 c1(C(=O)NC2CCC(N(C(c3cnc(C)s3)=O)C)C2)ccc(C2(F)COC2)cc1 Cc1cc(F)c(CC(=O)NCC2CN(C(=O)Cc3ccsn3)CCN2C)cc1F O=C(CC(=O)NCC1(F)CC(NC(=O)C2CC2)C1)NC(C1(CC(F)F)CC1)=O CC1OCCCC1C(=O)NCCN(C(=O)C=C(Cl)Cl)C1CC1 c1(C(N(C)CCN(C)C(C2(C3CCC3)CCC2)=O)=O)nnn2c1CSCC2 C1(CC)CN(C(=O)C(C)(C)F)CCC1NC(C1CCN(c2ccccc2)CC1)=O c1(NC(c2c(NC(c3c(OC)csc3)=O)cnc(F)c2)=O)ccc2ccccc2n1 CC1(CCNC(=O)Cc2cccc(F)c2)CCN(C(=O)CCc2cnccn2)C1 C1(C(c2n(CC(=C)C)nnn2)Nc2cnn(CCF)c2)CCC2(CC2)C1 C1(CC(=O)NCCC(O)CNC(C2(c3ccccc3)CC2(F)F)=O)CCOCC1 C(C(CNC(C1(C)CC1(Cl)Cl)=O)S(C)(=O)=O)NC(c1c(CC)n(C)nn1)=O N1(C(C(=Cc2cccs2)C)=O)CCN(C(=O)Cc2ccc(Cl)cc2F)C(C2CC2)C1 c1(OCC)ccnc2sc(C(N3CCC(CF)(NC(=O)C(C)SC)C3)=O)cc12 N1(C(c2ccc3cnccc3c2)C(=O)NCCSC)CC2CCC(C)(C1)C2(C)C C12(C(=O)NCCC(C)N(C(CCSC)=O)C)CC3CC(C1)C(F)(F)C(C3)C2 c1(OC)ccc2cccc(NC(=O)NCC(c3ccccc3C)C)c2c1 C1(CNC(C(CC)N(C)C)=O)CN(C(=O)Cc2ccc(OC)cc2Cl)CCCO1 CC(C(=O)N1CCC(O)(CCNC(C2CC(O)C2)=O)C1)C(F)F C(=O)(N=c1ccn(C2CCC2)[nH]1)c1c(C(C)NC(=O)CCCN(C)C)noc1 Cc1cccc(C(C(=O)NCC(F)F)N(C)CC2COCCO2)c1F C1(CCC)CN(C(=O)CN(C)CCO)CCN1C(C1CC(C)(C)CO1)=O C(=O)(CC(CC(C)C)NC(=O)C(O)CCSC)NC(CCC=C)C N1(C(c2c(OC)nsc2OC)=O)CCC2CN(C(C3CCOC3)=O)C2C1 N1(C(c2c(CC)n[nH]c2)=O)CC2CCOCC2(NC(=O)CCOC(C)C)C1 CCC(CCC(=O)NC1(C(N2CCC(C)(CCO)CC2)=O)CC1C)OC c1(C(N2CC(CC=C)(NC(=O)CCCc3cccs3)C2)=O)c(C)ncn1O N1(C(C(COC)C)=O)CCOC2(CCN(C(C3COC(=O)O3)=O)C2)C1 C(=O)(N1OC2CCC1CC2)n1c(C2CCCN(CC)C2C)nnc1S c1(CC(N2CCC(N(C(C=CCCCCC)=O)C)C2)=O)ccc(Br)c(F)c1 C(CCC1CCC1)(C(=O)N1CC(n2cnnn2)C1)NC(C1C(C)CC1)=O C(=O)(CC(CN(C)C)CC)NC(C1N(C(C(CC)=CCCC)=O)CCC1)(C)C C1(CN(C)C(C2CC2[N+](=O)[O-])=O)C2CN(C(=O)Cc3nccn3C)CC12 c1(CN2CC(F)(C(=O)NC3CC(C(=O)OC)C3)C2)c(C)cccc1Br N1(C(C(c2c(C)noc2C)CC)=O)CC(n2cc(CNC(N)=O)nn2)C(C)C1 N1(C(C2C(c3scc(C)c3)C2)=O)CCOCC1CNC(=O)CC1CC(C)(C)CO1 c1(C(N2C(C(=O)NCC(CC)CC)C(C)CC2)=O)cc(C)cc(F)c1 C1(C(C(=O)NC2C(NC(=O)CCCN3CCCC3)C2)O)CCCCCCC1 Cc1cc(N)cnc1C(N1CCCC1(C)C(=O)N(CCC(N)=O)C)=O c1(C(N2CCC(c3c(CNC(C4C(C(C)(F)F)C4)=O)c[nH]n3)C2)=O)cnn(C)c1Cl N1(C(CC(C(C)C)C)=O)CC2CCCC(N(C(=O)CCN3CCC3)C)C2C1 C1(C(C(C)=O)C)CCCCN1Cc1cccc(I)c1 c1(C(N(C)CC2CCCN(C(C3C(=C)C3)=O)C2)=O)sc(C#N)cc1Cl c1(SC)ccsc1C(=O)N(CCCCCNC(c1cc(C(F)F)no1)=O)C C(=O)(C1Cc2ccccc21)NC12CCC(C(N3C(C)(C(C)C)CC3)=O)(CC1)C2 C(=O)(CCCC(=O)NCC(CNC(=O)C(COC)OC)OC)NCC N1(C(CCC(=O)NCC)=O)CC(C)CN(C(c2conc2C2CCC2)=O)CC1C c1(CNC2(C)CN(Cc3ccc(OCC(=O)NC)cc3)C2)cc(F)c(F)c(F)c1 Cc1nc(=N)[nH]cc1C(=O)NCCC(C)CCNC(=O)C(C)(O)c1ccccn1 C1(NC(c2n(C)c(Cl)cn2)=O)CC12CCC(NC(=O)CN1CCNC(=O)C1)CC2 CCCCC(CNC(=O)CCc1ncccc1C)NC(C1CC2(CC2)CO1)=O C(=O)(C(C)(C)C(=O)NC1CC1CNC(c1sccc1C#N)=O)OC c1(C(N2CC3N(C(CC#N)=O)C(CC3)C2)=O)noc2cc(F)ccc12 C(=O)(CCCS(C)(=O)=O)NC(C)CCN(C)C(c1cn(C2CCC2O)nn1)=O c1(C(N(CC(C)(C)CNC(=O)CC2CC3C=CC2C3)CC)=O)c(F)cccc1F C1(CNC(CCN(S(C)(=O)=O)C)=O)CCC(F)(CNC(=O)Cn2cncn2)C1 c1(C(N(C2CCN(C(c3nccc(C)n3)=O)C2)C)=O)ccc2[nH]ccc2n1 N(C(=NCC1CC2(CC2)C1)N1CCCC(Cn2ccnn2)C1)C(C=C)C C1(CC(=O)NCC(C)=CC(=O)NCC2(C)CSC(C)=N2)CC(C)(C)CN1C C1(C(N2CCC(CC=C)(NC(=O)CCc3ccncc3)C2)=O)CC12CCSCC2 CC1=C(C)CC(C(=O)NCC(C2CCOC2)NC(=O)CSCC(F)F)CC1 Cc1cc(C(N2CC(O)(C(F)C(=O)NCc3nnnn3C)C2)=O)c(C)nn1 c1(C(N2C(C(N3CCC(OC)C3)=O)CC2)=O)ccc2nc(Br)sc2c1 C1(C(N(C2CCC(NC(c3cc(OC)n(C)n3)=O)CC2)C)=O)CCC(F)(F)CC1 N1(C(C(C)SC(F)(F)F)=O)CCC2C(CCN2C(=O)CCOCCOCCO)C1 N1(C(C2CC(C)OCC2)=O)CCCC(CNC(=O)C=Cc2cccs2)CC1 c1(CSCC(=O)NCCN(C(=O)CCCn2ccnn2)CC(C)O)nccn1C C1(C)(CNC(C(C)SC(C)C)=O)CC(NC(=O)Cn2nnnc2C(C)C)C1 CC1CN(C(=O)C=CI)CC(C)CN1C(c1cc(Cl)ncc1O)=O c1(C(=O)NC2(CNc3ccc(OC(C)C)nn3)COC2)ccc(C)nc1OC C(=O)(CC(CC1CC1)NC(c1cc(COC)no1)=O)NCC1(C=C)CCC1 N1(C(c2ncn(CC)c2)=O)CCC2C(C(=O)Nc3cn(C)nc3O)C2C1 N1(c2nccc(N3CCC(C(N4CCOCC4)=O)CC3)n2)CC2CCC(O)C2C1 c1(C(N2CC3C(CNC(c4cc(CC)no4)=O)C3C2)=O)cc2c[nH]nc2s1 c1(C(=O)NC2CN(C(c3nc(C#C)sc3)=O)CC2C)sc2cnccc2c1OC C1(C(N(C2CCN(C(=O)CC3CC3(C)C)C2)CC)=O)CC(F)(F)C1 CON1CCC(N(C(=O)CC2CCN(C(C3(C)CC4CC4C3)=O)C2)C)CC1 Cc1sc(O)nc1C(=O)NC(C)CC(C)NC(C1(C(F)F)CCCC1)=O Cc1csc(C#N)c1C(=O)NCC1CCCN1C(=O)C(c1ccnn1C)C N1(CC)CC(C(N2CCC(NC(=O)CCCc3ncco3)C(F)C2)=O)CCC1=O Cc1ccc2c(c1)C(C(=O)NC(C)CCCNC(=O)COc1ccccc1)C2 Cc1nn(CC(=O)NCC2CC2NC(c2ccn(CCF)n2)=O)cc1Br Cc1cc(C)n(CCC(N2CCOC(C(C)NC(=O)C=Cc3cnc[nH]3)C2)=O)n1 c1(C(=O)NC23C(CN(C(COCCOC)=O)C2)C3)cc(Br)c2ncccc2c1 N1(C(CC=C)=O)CC(C(=O)NC2CCCCC2)C2(CCC2)C1 n1(CCC)nc(C)c(C(N2C3CC2CN(C(c2ncc(F)cc2F)=O)C3)=O)c1C C(=O)(CC(C(F)(F)F)n1ccnc1)NCCCN(C(=O)Cc1cnoc1)C(C)C c1(CC)cc(C(N2CCC(N(C)C(c3cc(C)c(C)s3)=O)CC2)=O)ccc1O C1(C(=O)NC(CCC2CC2)C(=O)NCC2CC2(F)F)CC2CC1CC2O c1(OC)c(C(=O)NC2CC(CSC)C(O)C2)c(C)nn1C.c1(C(=O)N)ccc(C(N)=O)s1 c1(OC)c(F)ccc(F)c1C(=O)N(C)CC1(O)CCN(C(C2CC2C)=O)C1 C12(C(N3C4CN(C(C5CC(=C6CCC6)C5)=O)C(C4)C3)=O)CC3CC1C2C3(F)F N1(C(c2c(COC)ccs2)=O)CCC(n2cc(-c3cnc(C)o3)nn2)C(O)C1 C1(NC(CCC(=O)NCC)=O)CN(C(=O)C(C)OC2CCCCC2)CC1(C)C Cc1cc(C(N2CCN(C)CC2CNC(C2CCCS2)=O)=O)c(C)c(C)c1 N1(C(C2CCN(C(c3c(CC)cno3)=O)CC2)=O)CCCC(C)(N(C)C)C1 c1(C(=O)N(C2C(C)C2)C2CC2)cc(=O)n(C)c(O)n1.C1C(=O)N1.C12(CC1)CN2 N1(C(CCCOCC)=O)CC2(CC(NC(=O)C(c3cccn3C)O)CO2)C1 CCC(CC(C)C)C(=O)N1CC(CNC(C2(C)CS(=O)(=O)C2)=O)C2(CCC2)C1 C(=O)(CC(C)CNC(C1CCS(=O)CC1)=O)N(C1CSC1)CC#C N1(C(CCC)=O)CC(NC(=O)CCCOCc2ccccc2)C(SC)C1.C(C)OCC C1(CNC(C2C(=C)C2)=O)CCN(C(C2CCc3nncn3CC2)=O)CC1C1CC1 N1(C(c2c(Cl)c(C)n(C)n2)=O)CCC(NC(c2cccn2C2CC2)=O)C(CO)CC1 CCC(CN(C)C)C(=O)N1CCC(C(=O)NCC(=O)N(C)CC)C1C CC1SCCCC1C(=O)NCC1(C(N2CC(F)C2)=O)CCCCC1 C1(CN(C(C2C(C)CCC2)=O)C)CCCN(C(=O)CC(C)(C)c2ccccc2)C1 C(c1ccc(F)cc1)=CCC(=O)NC(C1CCN(C(C2ON=C(C)C2)=O)CC1)C c1(C(N2CCC(NC(C(C)Oc3cccc(F)c3)=O)C2)=O)csc2ccncc12 c1(CC(=O)NCC(CNC(c2c(C)cc(CC)o2)=O)F)ccc(F)cc1C(=O)O c1(N2CCC(C(N(OC)C)=O)C(C)C2)ccc(S(=O)(=O)N(CCO)C2CC2)cn1 c1(C(C(=O)NCCN(C(=O)C(C)CSc2ccccc2)CC)O)cccc(N)c1 C1(C(=O)NC(CC)(CNC(=O)CSCC(C)C)CC)Cc2ccccc2C1(C)C C(=O)(C1=CS(=O)(=O)CCC1)NC1C(C)(C)CCN(C(C2(C)CC2(Cl)Cl)=O)C1 C=C(Cl)CC1C(=O)N2CCC2(C)CO1.c1(C(=O)NCC2CC2)ncnn1CC c1(SC)ccc(C(=O)NCCC2(C(=O)NCCCN3CCC3)CCC2)o1 Cc1nc(C(=O)NC2CCCC2NC(C2CC(=O)NC(=O)N2)=O)ccc1[N+](=O)[O-] C(C(C)(C)CNC(=O)C(O)Cn1cncn1)N(C)C(C1CCSC1)=O Cc1n[nH]c2cc(C(=O)NC3CCCCC3NC(C3(C)CCCS3)=O)ncc12 S(=O)(=O)(c1ccccn1)N1CCN(C(c2cccc(SC)c2)=O)C(C(F)(F)F)C1 C1(C(N(CC(C)OCC)C)=O)CC=CC(n2cc(CC(C)C)nn2)C1 CC(C)(O)C(C(=O)NCc1n[nH]cc1C1CC1)NC(=O)CC1CCOC1=O C1(C(N2CC(C(C)NC(C=C(C)C)=O)OCC2)=O)CC2(CCCCC2)S1(=O)=O C1(NC(=O)CCc2ccc(O)cc2)CS(=O)(=O)CC1NC(C1(CO)CCC1)=O c1(CC(=O)NCCN2CCN(C(C3CCC3)=O)CC2)c[nH]c2c(Br)cccc12 N1(C(CC2CC(=C)C2)=O)CC(O)CCC1C(=O)N(CC)CC1CN(C)CCN1C c1(CCC(N2CC(CNC(c3c(OC)ccnc3)=O)C2)=O)ccc(F)cc1F C1(C(N2CCC2CC2CCCC2)=O)CCC(O)CN1C(=O)C=CC1CCC1 CN1CCC=C(c2ccco2)CN(C(=O)OCc2ccc(Cl)c(S(N)(=O)=O)c2)C1 c1(OC)nccc(NC(N2CCCC(c3nc(C)c(C)s3)C2)=O)c1Br C(=O)(CCCC(C)C)NC1C(CN(C(c2c(CC)n(C)nn2)=O)C)CCC1 C1(C(=O)NCc2nnc(CC)s2)CC(C)CN(C(C2OC3CCC2C3)=O)C1 c1(C(=O)NC2(C#N)CCN(C(c3ccno3)=O)C2)c(F)cc(Br)cc1Cl C(CC(C)C(=O)NC(C1CC1C(=O)N(CC)CC12CCC(CC1)C2)C)=CC c1(C(C)(C)C)ccc(C(C)(C)NC(c2ccc(CF)cc2)=O)cc1 C(=O)(C1(C)CCCc2ccccc21)NC1CN(C(C2(SCC)CC2)=O)CC1C c1(CCC(=O)NC2CCN(C(c3c(SC)nccn3)=O)CC2)c(C)ncnc1O C1(O)(CNC(C2C(=C)CC2)=O)CCN(C(c2c(C)noc2C(F)(F)F)=O)C1 C1(C(=O)NC(C(C)C)C2CC2)CSCCN1C(=O)Cn1ccccc1=O C12(NC(c3c(CC)nns3)=O)CCN(C(c3cnc(Cl)c(N)c3)=O)CC1C2 C12(NC(C3CC4(C3)CC3(CCC3)C4)=O)CCCCCC1N(C(=O)C=CCF)CC2 C1CCC2=C3NC(=NCCC(CCOC)C3)OC2=NC2CC3CCC2C13 c1(C(=O)NC2CC(NC(C)=O)C2)ccc(Cl)c(Cl)c1N c1(C(N2CC(CC(C)NC(c3cnn[nH]3)=O)C2)=O)cc(Cl)c(Br)[nH]1 C(=O)(C1=CS(=O)(=O)CCC1)NCC1C(C)CCN(C(=O)Cc2ccn(C)n2)C1 C1(NC(C2(CC(C)=O)CC2)=O)COCC1CNC(=O)CC1(C2CC2)CC1 Cc1ncc(C(=O)NC23CCC2CN(C(=O)Cc2cnns2)C3)c(C(C)C)n1 CCC(=O)CCC(=O)N(C(C)C(=O)NCc1ccc(F)c(C)c1)CC O=C(CCCC1CC1)NCCCN(CCO)C(c1cnc(-c2ccccc2)o1)=O C(c1ccc(C(N)=O)o1)=CC(=O)N(CC(CC)N)C.C1(C(=O)N)(C(=O)OC)CC1C CCCCC(O)C(C)C(=O)NC1CC(C(=O)NCC23CCCC2C3)=CC1O C(=O)(C(C)(C)CC(=O)N1CC(C(=O)NC(C)(C)CCCF)CC1(C)C)OC c1(C(=O)NCC=C(C(=O)NC(CC)C)C)cncc(CO)c1 CC1CC=CCC1C(=O)NCC1CCC(NC(=O)NCCOC(C)(C)C)C1 C1(C(=O)NCC(CO)NC(c2c(CC)nc[nH]2)=O)CC(C(C)(C)C)=NO1 CC1CN(C(C2Cc3cccc(C)c3O2)=O)CCC1N=c1ccnc(Cl)[nH]1 C(CC(C(C)(C)C)NC(C1(C(=O)OC)CC1)=O)N(C(CC1(CC(=O)OC)CC1)=O)C c1(C(=O)NC2(CO)CN(C(C(c3cn(C)nc3)O)=O)C2)cccc2nc(O)[nH]c12 CN=c1nc(N2CCN(CCOC)CC2)[nH]c(=NCCC2COCC(C)O2)[nH]1 c1(CCC(=O)NC(C)CN(C2CC2)Cc2ccsc2)nc(O)c2cnn(C)c2n1 c1(Cn2cc(C(C3CC3)NC(C3C(=O)NCCC3)=O)nn2)ccc(Cl)cc1Br N1(C(C)C)C2CCC1CC(c1nnnn1C)(NCCc1c[nH]c3cnccc13)C2 CC(CNC(c1cc(Cl)ns1)=O)C(=O)NCC1CSCCO1 C(C)(CC(=O)N(CC=C)OC)NC(C)=O.C1C(=O)N1CC#C C(=O)(C(O)CCC(C)C)NC(C(=O)NCC(=C)C)CCC1CC1 N1(C(CCS(C)(=O)=O)=O)CCC2(COC(CNC(c3c(Cl)ccnc3F)=O)C2)C1 c1(C(N2C(C)CCC2CNC(=O)C(C)(C)C(F)F)=O)nn(C)cc1[N+](=O)[O-] CC1(C)C=C(C(=O)NCCOC2CN(C(=O)CC3CC(C)(C)C(=O)N3)C2)C1 N1(C(C2CCC(CC)O2)=O)CC(NC(=O)Cn2ccc(C)c2)C2CCCC12 N1(N(c2cnccc2C(F)(F)F)C)CC2(C1)CN(C(=O)C(C)(C)C1CCC1)C2.C(C)=O CCCCC(Cc1ccccc1)NC(=O)NC(c1ccccc1)C(=O)OC c1(C(=O)NC2CC(C)CN(C(=O)C=C(Cl)Cl)C2)oc2ccccc2c1Cl c1(C(N2C(CO)CC(NC(C(C)CO)=O)C2)=O)ccn2c(Br)cnc2c1 c1(C(C(=O)NCCCN(C(CC)=O)C2CC2)O)cc(F)c(F)c(F)c1 c1(CNC(C(CNC(CSCCC)=O)(C)CC)=O)c[nH]c2c1CCCC2 N1(C(c2cnc(C)nc2)=O)CCC2(C1)CN(C(=O)CC(C)(C)CN(C)C)CCO2 c1(C(=O)NC2C(NC(C3C(C=C)CC3)=O)CCCC2)ncn2ccccc12 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CC2C(CNC(C(C)O)=O)C2C1 c1(C(=O)NC(C2CCN(C(C(C(C)C)(C)O)=O)CC2)C)cnc2cccnc2c1 CC1(C(=O)NCCn2cc(C(=O)NCC(Cl)=CCl)cn2)CC(O)C1 c1(C(N2CCC(O)(CNC(C=CSC)=O)C2)=O)cnc(=NCCF)[nH]c1 CN1C(=O)OCC1C(N1CC2CC1C2C(N1CCCC1C(C)(C)C)=O)=O S(=O)(=O)(c1ccc2c(c1)OCCO2)NC12CC(C(N3Cc4ccccc4C3)=O)(C1)C2 N1(C(Cc2ccc(C)cc2)=O)CC(F)(F)CC1C(=O)NCC1(C)CC2CCC1C2 C(=O)(C(c1cncs1)N(CCCO)C(C)(C)C)NCCC1(C)CC1 c1(OC)ccc(C(=O)Nc2ccnc(-c3cncc(O)c3)c2)c(F)c1F CC1C(C(N2CC(CC34CC(C3)C4)C2)=O)CCCN1C(c1ccc(=N)[nH]c1)=O c1(C(=O)NC2CC(CNC(C(C(COC)C)C)=O)C2)c(O)ccc(F)c1Br CC(C)C(CNC(=O)C=Cc1ccc[nH]1)C(=O)NCCc1cncn1C N1(C(C2C(=C)CC2)=O)CCN(C(C2CN3CCN2CC3)=O)CC1CCO N1(C(C2(C)C(C)CCC2)=O)Cc2ccc(CNC(c3ccc(O)nc3)=O)cc2C1 C1(C(=O)NC2CC(C)C2)CC(F)C(=O)N1.c1(SC(=O)C2CC2)ccncc1.O=C1CC2(CC2)N1 Cn1nc(C(=O)NC2CC2NC(C2(N(C)C)CCOCC2)=O)cc1C(C)(C)C C1(O)(CN(C)C(c2n[nH]cc2Cl)=O)CN(C(=O)C(C)(O)C2CC2)C1 c1(CCC(=O)NCC2CCN(C(=O)C(F)CC3CCCC3)C2)ccccc1Cl N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)C1CNC(=O)CCC(C)(C)F C(=O)(CC(C)C(=O)OC)NC(C(=O)NC(CCC)C1CCCC1)Cn1cncn1 CC(C)C(C(=O)N1CCCC1)NC(=O)CC(C)O C1(CNC2(c3n(C(CC)C)nnn3)CCOC2)CCNCC1.C(=O)(NC)NC C1(C(N(C2CCC(NC(CCCCN(C)C)=O)CC2)C)=O)CC12CCCOC2 CC(C)(C)C(CNC(C1COCCN1C(C1CCSC1)=O)=O)CO C=C(C)CC(=O)NCCN(C(=O)C(c1cc(Br)co1)=O)CCOCCO N1(C(C)C(=O)Nc2ccc(OCF)cc2)CCC(O)C(O)C1 n1(CC)cc(C(=O)NCCc2ocnc2CNC(c2cnc(C)s2)=O)c(C)n1 c1(NS(c2n(CCOC)ncc2)(=O)=O)nc(C(F)(F)F)ccc1C#N CC1CN(C(C2(N(C)C)CCCC2)=O)CCC1C(=O)N(CC(F)(F)Cl)C c1(C(C(=O)NCCN(C)C(C2CC=CCC2)=O)NC(=O)C2CC2)cnn(C)c1 c1(NC(=O)NOCC(C(C)OCC)C)cc(Cl)cc(Cl)c1 C(=O)(CC(C)(F)F)N(C1(CCO)CCCC1)C(C(C)C)C Cc1nc(O)sc1C(=O)N(CC(C)(C)NC(c1ccc(CO)nc1)=O)C Cc1cc(C)c(C(=O)NCC2(O)CN(C(=O)C(=Cc3cn(C)cn3)F)C2)[nH]1 C1(C2CN(C(=O)Cn3cccc(C)c3=O)C2)(NC(CCn2c(C)ncc2)=O)CC1 C=CC(C(=O)NC1CC(CC(=O)NCC(CO)OC)C1)OC C12(CNC(C3=CC(C)(CC)C3)=O)CCCC1N(C(c1csc(C(F)F)n1)=O)CC2 C1(C(=O)NCC(CC)NC(=O)C=Cc2scnc2C)CCC(O)CN1C C1(CC)CCOC1C(=O)NC1CC(C)(NC(=O)CCc2ccoc2)C1 N1(C(CC2ON=C(CC)C2)=O)CCC2CC12C(=O)N(CC(O)C1CCC1)C c1(OC)ccc(-n2nnnc2C2(NCc3nccs3)CCCC2CCF)cc1Cl c1(C(N2CCC(C(=O)NC(CC#C)CC)C2C)=O)cccc(C#N)c1 c1(N(C)CC2CCCN(C(c3cnc(C)[nH]3)=O)C2)ncnc(C)c1C#N N1(C(C(C)OCCOC)=O)CC2(CCCN(C(c3cnc4nccn4c3)=O)C2)C1 C1(NC(C(C)=C(C)C)=O)CC(CNC(=O)C=Cc2cnc[nH]2)C12CCC2 N1(C(C(C)=C(CC)C)=O)CCN(C(=O)CP(C)(C)=O)CC1c1ccnn1C N1(C(c2n(C)cc(Cl)c2)=O)CCC2(CCCN(C(C3CC(F)(CO)C3)=O)C2)C1 C12(C(=O)OCC)CC(CO1)N(C(=O)C(C1(O)CN(C(=O)NC(C)(C)C)C1)F)C2 S(=O)(=O)(c1cccc(=NCC(C)N(C)C2CC2)[nH]1)N1CCC(CC)C1 Cc1cc(Br)cnc1C(N1CCC(C)(NC(=O)CN2CCOCC2)CC1)=O N1(C(C2CCCOCC2)=O)CC23CCCCC2(C1)CN(C(C1CCCOC1)=O)C3 CCC(O)C(F)(F)C(=O)NCC1CCCN1C(C1CC(CF)C1)=O C(CCC(=O)NC(C)CNC(c1cnc(CC(C)C)o1)=O)N(CC(=O)NCC)C C1(NC(CCOCCC)=O)CCCC1CNC(=O)Cc1cnns1 CCC(Cc1ccccc1)CC(=O)N(CC(C)NC(=O)C(C)(C)n1cccn1)C N1(C(CCc2nc(=N)[nH][nH]2)=O)CCCC(CO)(CNC(C23CCC(C2)C3)=O)C1 C1(Nc2c(Cl)cnc(C(C)C)n2)CC2CCC1N(C(c1ncccc1Cl)=O)C2 O=C1CCC(n2ccnc2-c2cccc(-c3cccc(Cl)c3)c2)CN1 CCN=c1[nH]c(C)c(C(N2CC3CCC2C(NC(C2C4CCCC24)=O)C3)=O)s1 C1(CCNC(C2CC3(CCCC3)C2)=O)CC(F)(F)CN1C(=O)C=CCF C1(C(=O)NC(CC)(CNC(=O)C(c2cccnc2)O)CC)CN2CCC1CC2 N#Cc1nc(Cl)ccc1NC(C1CSCCN1Cc1ccc([N+](=O)[O-])o1)=O N1(C(C2CC3(CC(=O)N3)C2)=O)CC(C2CCN(C(C3(CO)CCC3)=O)CC2)C1 N1(C(CSCCCC)=O)CC(NC(=O)CC(CC)C2CCC2)C2(CCOCC2)C1 c1(OC)ncc(C(=O)NCC2(F)CC(NC(c3csc(Cl)c3)=O)C2)s1 CC1(C)COC(CNC(C2(CNC(C3CCCC3(C)C)=O)CC2)=O)C1 c1(CC)cc(C(N2CCN(C(=O)CC(O)CN(C)C)CC2C)=O)ccc1F Cn1ccc2cccc(C(N3CCC(CO)(NC(=O)Cn4cccn4)C3)=O)c12 C=CC1(CNC(C2CC2C2CN(C(=O)CSC(F)(F)F)C2)=O)CCOCC1 c1(C(=O)NCC(C)(C2CC2)NC(C(C=C=C)C)=O)ccc(OC)nc1Cl CCCCCCCCOCC(=O)NC1CN2CCC1(CSc1ccccc1)C2 c1(N2CCN(C(c3c(OC)csc3)=O)C3(C2)CC3)ncnc2cc(F)ccc12 N1(C(c2conc2C(F)(F)F)=O)CCCCC12CC(NC(C1(F)CCOC1)=O)C2 CN1CCCCC1C(=O)NCC(CO)NC(=O)C(C)(C)n1cc(Br)cn1 c1(C(NC(=NC)NCCc2ccccc2)C2(CCC)CC2)ccc2c(c1)OCO2 CC1CCN(C(=O)C=CC2CC2)CC1NC(=O)CCC1CCCO1 C1(NC(C2CC2[N+](=O)[O-])=O)CCC(CNC(C2(O)CC2)=O)CC1 CC1(C#CC(=O)NC2C=CC(CNC(c3coc(Br)n3)=O)C2)CCCO1 N1(C(C=CCNC(=O)CCn2ccnc2)=O)CCn2nccc21 c1(NC(=O)CC2CCN(C(c3cccc(F)c3I)=O)C2)ncnc2[nH]c(Br)nc12 CCCCS(=O)c1ccc(CC(=O)N2CCC2CCCCCO)cc1 Cc1ccc(N2CCN(C(C)C(=O)Nc3ccc(F)cc3Br)C(C)C2)cc1C N1(C(CSCCC)=O)CCN(C(c2ccnn2CC(C)C)=O)CC1C(C)C C1(COC(N(CCOc2ccccc2NS(N)(=O)=O)CC)=O)CC(=O)NC(C)C1 C(=O)(C1=COCCC1)N1CCC(NC(C(C)(CNC(=O)C(C)C)OC)=O)C1 Cc1nc(Cl)ncc1NC(C1C=CCN1C(C1CCCS1)=O)=O c1(OC)cc(OC)c2c(c1)N(C(=O)C(N1CC(C)N(C)C(C)C1)=O)CCC2 Cn1cccc1C(=O)NCC1(CNC(C2CCC=CO2)=O)CC1 CC(C)C(C)CC(=O)Nc1cc(O)nc(F)c1.C12CN(C1)C(=O)CO2 C1(C(CNC(CC2N(C(C)=O)CCC2)=O)(C)C)CCCCN1C(=O)C(=O)N(C)C c1(C(=O)NC(C2CCN(C(=O)C(O)c3ccsc3)C2)(C)C)cccc(F)c1F N1(C(c2ccnc(CN(C)C)c2)C(=O)NCCOC)CCC(C)(NC(C)=O)CC1 Cc1cnc(CCNC(C2CCCC2CNC(c2cscc2C)=O)=O)nc1 CCC(C)(C)CCCC(=O)NCC1CCN1C(c1cncc2ccsc12)=O [nH]1nc(C)c(C(=O)NCCC=O)c1C.C1(COC)CC1NC(=O)CNC=O.OC C(=O)(C(O)CC(N)=O)N1C(C(=O)NCC(CSC)(C)C)CSCC1 C(=O)(C(O)C(C)CC)NC(c1cnn(C)c1)C(=O)NCCCCCC=C c1(C(=O)NCC2(C)CCN(C(C3CC(C)(F)C3)=O)C2)ccc2c(c1)OCCO2 c1(C(=O)NCCN(C(C2CC(O)C(F)C2)=O)C2CC2)cc2c(cc1O)OCO2 C1(C(N2CC(NC(C3N(C(C(C)(C)C)=O)CSC3)=O)C2)=O)CCc2ncccc2C1 N1(C(CCC(=O)NCCC)=O)CC2(CCC2)CC1C(N1CCC1CC)=O C1(C(=O)NC2(COC)CN(C(c3ccncc3C)=O)C2)(COC)CCOCC1 Cc1nccnc1CCNC(=O)C(C)(C)NC(c1n[nH]c(O)n1)=O C=CCCCC(C)(C)C(=O)NCCC1(NC(=O)C(C)n2cnnn2)CC1 N1(C(C2(COC)CCCCO2)=O)CCC(C)(CNC(=O)CC2CC2)CC1 N1(C(C2(CSC)CC2)=O)CCOC(CN(C(=O)Cc2ccon2)C)C1 C#Cc1cccc(CC(N2C(CC(=O)N(C(C)CSC)C)C3CCCC23)=O)c1 N1(c2nccc(C)n2)CCN(C(C23CC(CN2C2CC2)C3)=O)CC1C N1(C(C2(OC)CCC2c2cccc(C)c2)=O)CCN(C(=O)CCF)C(CO)C1 c1(OC)ccnc(C(N2CC(CO)(NC(c3ccc(SC)cc3)=O)C2)=O)c1 N1(C(=O)Cc2csnn2)CCC2CC12C(=O)NCCCc1ccsc1 c1(C(=O)NC(C(=O)NC2CCN(CC)C2)C2(O)CCC2)ccc(CF)cc1 N1(C(c2ccc(C)cc2N)=O)CCCC2CN(C(=O)CN(C3CCC3)C)CCC12 C1(n2c(C(c3cccc(C)c3)NCCO)nnn2)CCC(F)(F)CC1.C1CCCC1 C1(C(N2CCC(OCC(=O)NC3(C)CC(O)C3)C2)=O)CC2CCC1CC2 C1(C#N)(C(N(C)CCOCCNC(c2coc(C(N)=O)c2)=O)=O)CCC(=O)CC1 C1(NC(C2(COC)COC2)=O)CCCC(CC(=O)NCCC(C)(C)CC)C1 C1(NC(CC2(CSC)CC2)=O)CCCCC1CNC(=O)C(c1ccc(C)s1)C CC1=C(C(=O)NC(CC2CC2)CC(=O)N(C2CCCNC2=O)C)CC1 CC(C)(C(=O)NCC1CC(O)(CNC(=O)C=Cc2ccc(O)cc2)C1)C(F)F N1(C(Cc2c(C)noc2C)=O)CCC2(CC2C(=O)NC2CCC(C)(C)CC2)C1 C=C(C)C(C)(O)C(=O)NCCC(C)N(C(=O)CCOC1CC1)C C12(C(=O)NC(CN(C(c3nc(C(C)C)sc3)=O)C)C)CCC(=O)N1CCS2 CON=CC(=O)NCC1(CC(=O)N(CCCF)C)CC1 c1(C2C(C(N3CC(NC(CCCC=C)=O)C(C)C3)=O)C2)ccc(C)c(C)c1 C1(C(N2CCCC(NC(CSC)=O)C2)=O)CC(=O)c2cc(Cl)ccc2O1 C1(NC(CCN(C(c2cnc(CC)s2)=O)C)=O)COCCC1CC C(=O)(CS(=O)(=O)CC(=O)OC)N1CC(NC(CC(CC)(F)F)=O)C(C)CC1 C(C)(C(CO)NC(=O)CC1(C)CC1)NC(CN(CCc1ccccc1)CC)=O CC1=C(CNC(CCC(F)Cn2cc(CC(C)O)nn2)=O)C(C)CCC1 CC1(C(=O)Oc2ccccc2)CC12CCN(C(=O)NCCc1ccccn1)CC2 c1(CC(=O)NC(CN2CCN(C(C3(C(C)=O)CC3)=O)CC2)C)cc(C)cc(F)c1 CC(C)(C)CCCCC(=O)NC1CC2CN(C(C3(C4CC4)CCCO3)=O)CC2C1 C=CCC(CC)C(=O)N1CCC(CNC(C2CC3(CCO2)CC3)=O)C(O)C1 c1(C(=O)NCc2cn(C3C(OCC)COC3)nn2)ccnc(-c2nccs2)n1 C(=O)(C1=NNC(=O)CC1)NCC(=C)CCNC(=O)CCCOCCOCC C=C(C)CCCC(=O)NC(C)CC(C)NC(c1ccc(-n2ccnc2O)cc1)=O CC1CC(C)(C(=O)N(C)CC2(NC(=O)C(C)(C)F)CC2)CCO1 N1(C(C)=O)CCCC(C(N2C(CNC(=O)CC3CC3(C)C)CC3CC23)=O)C1 CC(C)(C)C(CNC(c1cc([N+](=O)[O-])n[nH]1)=O)C(=O)NC1CCC(C(N)=O)C1 C(=O)(C(CO)C(C)(C)C)NCC1N(C(CN2CCC(C)CC2)=O)CC(O)C1 C1(CNC(C2C(OCCOC)CC2)=O)(O)CCCC1.C(=O)(C(CC)NC1CC1)N C(C(=O)N1CCCC(CNC(=O)C(=Cc2cnc[nH]2)C)C1)(C(C)C)OC c1(C(N2CC(NC(c3nccc(N)c3)=O)C2)=O)c(F)ccc(Br)c1F N1(C(C(C)C2CCCO2)=O)Cc2occ(C(=O)NC(C)(C)CC3CCC3)c2C1 CC1(C)CCCOC1C(=O)NC1CN(C(=O)CCC2CC2(F)F)CC1(C)C c1(OC)cccc2c1OCC(C(N1CCCCCC1CCO)=O)C2 C(=O)(C(C)C(C)(F)F)NCC(C)NC(C(C(C)C)O)=O C1(C(=O)NC(C)Cc2cn[nH]c2)COC(CNC(=O)Cc2ccc(Cl)s2)C1 C=CC1OCCC1NC(c1cc(CNC(C2(C#N)CCOC2)=O)on1)=O c1(C(N2CC3C(CNC(c4c(C)cccc4)=O)(C3)C2)=O)cncc(O)c1Cl C1(CNC(C2(OC)CCSCC2)=O)CCC(C)CN1C(=O)CSCC(C)C c1(C(=O)NCCC(N)=O)ccc(-c2cn(CCO)nn2)cn1 N1(C(CCN(CC)CC)=O)CC(NC(c2ccc(C)c(OC)c2)=O)CC1(C)CC c1(C(=O)NC2CN(C(C(CC)CCOC)=O)CC2C)ccc(S(C)(=O)=O)cc1N c1(C(=O)NCC(CN(C(C2(CCC#C)CCC2)=O)C)C)ccn(C(C)C)c(=O)c1 c1(C(N2C3C(CNC(c4cnc(O)s4)=O)C(C3)C2)=O)cc(Cl)ccc1Cl N1(C(C(CCC)OC)=O)CCN(C(c2ccc(Cl)cc2C)=O)C(CF)C1 Cn1ccc(C=CC(=O)NC2CC2NC(c2ccc(Cl)o2)=O)c1 CC(N=c1ccnc(N2CCC(CC#N)C(F)(F)CC2)[nH]1)c1ccc(Br)cn1 c1(-n2c(C(=O)NCC(C)(C3CCC3)NC(=O)CO)cnc2)ccccc1F N1(C(CCC)=O)CC2CCCC(CNC(c3ccc[nH]3)C3CCCC3)C2C1 N1(C(=O)NCC(CC#C)C2CC2)Cc2cccc(Br)c2CC1C(=O)OCC O(N(C)C1CCc2ccc(OC)cc21)CC(=O)OCC C1(C(N(CCNC(C(C(C)C)NC(=O)OC(C)C)=O)C)=O)CC2CCC1CC2 c1(C(=O)NC(CN(C(c2ccn(CCCC)n2)=O)C)CC)cccc(C)c1CC CN1CC=C(CC(=O)NCC2CC2C(=O)NCCCc2cccs2)CC1 CCC(CCCC(=O)NCC(C)CC1CC1)NC(c1sccc1C)=O CC1CC(C)CN(Cc2ccc(NC(=O)N(CCCC(C)(C)N(C)C)C)cc2)C1 N1(C(C(C=C)(C)C)=O)CCC(C(F)(F)F)C(NC(=O)C(c2cncn2C)O)C1 C1(CN(C(CC2(COCC)CC2)=O)C)CCCCN1C(=O)C(C)CNC(C)=O Cc1nccc(N2CCN(CCN(C(=O)CCCc3cnn[nH]3)C)CC2)n1 C1(C)(C(N2CCC(OC3CN(CC4ON=C(C)C4)C3)C2)=O)CCCCNC1=O C1(C(=O)NC2C(C)(C)C2C(=O)NCC(F)(F)F)CCC2(CC2)C1 C1(C(=O)NC(C(C)NC(c2ccc[nH]2)=O)CO)CC(C)(C)C(C)(C)C1 C(N1CCCC(C)(C)C1)N1C(=O)CC(C2CN(CCCCCC)C2)C1 Cc1cc(=NC2CCCC2C#N)[nH]c(=NCc2cccc(S(C)(=O)=O)c2)[nH]1 N1(C(c2c(OCC)scc2)=O)CCC2CC1CN(C(C1COCC(C)(C)O1)=O)C2 C(=O)(C(C(C)O)NC(c1ccc(OC)o1)=O)N(CC)CC1CCCO1 c1(C(=O)NC2CCCN(C(CC(CC)OC)=O)C2C)cnc2[nH]c(O)nc2c1 CC1C(NC(c2nn[nH]c2Cl)=O)CCCN1C(=O)CSCc1ncc[nH]1 C1(C(=O)NC(CCOC)CNC(C2CC(=C(F)F)C2)=O)(C(C)C)CCN(C)CC1 C1(C2(NC(c3n[nH]cc3C3CCC3)=O)CC2)CCCN1C(=O)CC1(O)CCCC1 c1(CC(=O)NCC(N(C(CC=C(C)C)=O)C)C2CC2)coc2ccc(C)cc12 N1(C(c2c(C(C)C)occ2)=O)CC(NC(c2cncc(N)n2)=O)C(C)C1 C1(NC(C(C)SC(C)C)=O)CC2C1CCN2C(c1ccnc(S)c1)=O C(=O)(C(=O)CCC(C)C)N(C1(C(=O)NCCCOC(=O)NC)CC1)C N1(C(C2C(COC)C2)=O)CC(CO)(NC(=O)Cn2ccnc2C(C)C)C1 C1(C(=O)NC2C(NC(C3(C)CCC3)=O)CCCC2)OCC2CCCCC12 Cc1cc(C(N2CCC2CNC(c2cc(Cl)no2)=O)=O)nnc1C C1(OC)(CNC(C2(C#N)CCCO2)=O)CCN(C(C2(C)CNC(=O)N2)=O)C1 C(=O)(C1=CCS(=O)(=O)C1)NC(CNC(C(CC)(C)C#N)=O)C1CC1 c1(-c2cc(C(=O)NCC(C3CCC3)NC(CCSCC)=O)no2)cccc(Cl)c1 N1(C(=O)Cn2ccnn2)CCCC(O)(CNC(C2(c3ccncc3Cl)CC2)=O)CC1 c1(CC(=O)NCC(Cn2cc(-c3ccc(CC)s3)nn2)(C)C)cc(Br)cn1C C(=O)(C1CCc2nccn21)NC(C)(CO)C(=O)NC1COCC1CO C1(CNC(=O)Cn2cccn2)CN(C(c2ccn3cccc3c2)=O)C2(CCC2)C1 N1(C(CC2(COC)CC2)=O)CC(NC(c2c(C3CC3)cnn2C)=O)C(SC)C1 N1(C(C2(OCC)CC2)=O)CCC(C)C(NC(=O)CNC(c2ncccc2O)=O)C1 c1(C(N(CCN(C(C(C)OCCOCC)=O)C)C)=O)cc(C(F)(F)F)nc(O)c1 c1(C(=O)NCC2N(C(C(C)SC(C)C)=O)C3C(C2)C3)ccnn2ccnc12 C1(=O)CCCCCO1.C12(C(=O)OC)CC1CN(C(=O)OCc1cccc(Br)n1)C2 C(C)(CCC(=O)c1ccc(CN2CCCCC2C)cc1)N(C(=O)C(=O)NC)CC C1(CCC)(C(=O)NC2CC2NC(c2ccccc2OC(F)F)=O)CCNC1=O c1(C(C(=O)NCC(CC)NC(=O)CCNC(=O)CC(C)C)C)c(C)n[nH]c1C Cc1nccn1CCCC(=O)NCC(C)CN(C(=O)CCN1CCCCC1)C C1(NC(C(C(CC)C)O)=O)CCSC12CN(C(c1cnc(N)c(N)c1)=O)C2 C(=O)(CCCCCNC(c1cc(F)ccc1F)=O)N1CCC(O)(CC)C1 CCC(CC(=O)N1CC2CCOC2(CNC(C2(CCF)CC2)=O)C1)C(C)(C)C c1(C(=O)NC2C(NC(c3cn(C(C)(C)C)nc3)=O)C2)cccc(N)c1Br C1(C(=O)NC2(CC=C)CN(C(=O)CCc3ncc[nH]3)C2)CCCOC1C Cc1coc(C(c2nnnn2CSc2ccccc2)NC2(C)CC2(C)C)c1 C=CCC(CC)C(=O)NCC1(C(=O)NCC2(COC)CC2)CC1 CC1CN(C(N2CCOCC2C2CC2)=O)CC(=O)N1 C(=O)(C(C)(C)C(C)(F)F)NC1C=CC(C(N(CC(C)OC)C)=O)C1 CN1CCCC2CN(C(C3CC4(C3)CC3(CNC3)C4)=O)CCC12 c1(C(N(C(CNC(=O)Cc2cccs2)C2CC2)C)=O)ccc([N+](=O)[O-])c(O)c1 N1(C(CC(=C=C)C)=O)C2CCCC1CN(C(C1CCC(=O)N(CC)C1)=O)CC2 c1(C(=O)NCCC(=C)CNC(c2cnoc2CC)=O)c(Br)c(C)nn1C c1(C(=O)NC(C)C(=O)NC(c2nnc(S)o2)C)ccc(S(=O)(=O)N(C)C)cc1 N1(C(c2c(C)nn(-c3ccncc3)c2)=O)CCCC(NC(=O)CC2CCC2)CC1 Cc1[nH]cc(C(N2CCCC(C)(CNC(c3ccc[nH]3)=O)C2)=O)c(=O)c1Cl O(NC(=O)C(C)(C)CCNC(c1c[nH]cc1C)=O)C(C=C)C CCC(C(=O)NC(CNC(c1ncccn1)=O)C(C)C)C(C)C C1(C(N2CC(C3(NC(=O)C4=CCCCC4)CC3)C2)=O)CC12CCc1ccccc12 C12(NC(c3cncc(C(=O)OC)c3)=O)CCCN(C(=O)C(O)c3ccsc3)C1C2 c1(OC)ccc(C=CC(=O)NCCCCN=[N+]=[N-])c(OC)c1 CCC(O)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)C(C)(C)c2ccccn2)C1 CC1CN(C(=O)C=C(C2CC2)C2CC2)CC(CCNC(c2cc(Cl)c[nH]2)=O)O1 Cc1cc([N+](=O)[O-])cc(C(N2CC(NC(=O)CSc3cccs3)CC2(C)C)=O)n1 CC1(C(N2CC3(C2)CN(C(=O)CSc2cccs2)C3)=O)Cc2ccccc2N1 C1(C(=O)Nc2c(O)ncnc2O)C2CC(F)C(C2)N1C(=O)Cc1ccco1 c1(C(=O)OC2C(c3cn(CC)nc3)C2)c(OC)cccc1C(C)C Cc1cc(C(F)F)nn1CC(=O)NCC(C)NC(c1c(Cl)cnn1C(C)C)=O c1(C(=O)NC(C)C(C)NC(c2ccn(CCO)c(=O)c2)=O)c(F)cc(F)cc1Cl C(N=c1nc(N2C3CCC2CC(O)C3)c2c([nH]1)CSC2)c1c(CC)noc1C c1(CNC(C(C)CF)=O)cccc(CNC(C2CSC2)=O)c1 CC1(CNC(C2CSCCS2)=O)CCN(C(c2cnccc2Cl)=O)C1 n1(CC(=O)NC2(C)CCN(C(C3C(C)=C3)=O)C2)ccc2cc(F)ccc12 c1(C(N(CCCN(C)C(C2(C)CCCCO2)=O)C)=O)cccc2nsnc12 N1(N2c3c(cc(C)c(Br)c3)CC2)CCc2c(cccc2[N+](=O)[O-])C1.C C1(NC(CCCC(=C)C)=O)CC2CN(C(=O)CC3CCC(C)(O)CC3)CC2C1 C12(CCOCC1)C(C)C(=O)N2.C1(N(C(=O)C=CCN)C)CCOC1=O c1(N)ccc(F)cc1Br.c1(C2(C)CC2)ccc(C2(C(=O)O)CC2)cc1 C1(Nc2cc[nH]c2)CN(C(C2CCN(c3ccc(Cl)cc3)CC2)=O)CC12CC2 N1(CC(=O)NCC2(O)CC(NC(c3n(C)ccc3)=O)C2)CC(=O)NC1=O N1(C(CN2CCC(OC)C2)=O)CC(OC)CC1(C)COC(F)F.C(=O)(CN(C)C)N C(=O)(C1CCCc2nn[nH]c21)N1CC2C(NC(C#CC3(C)CC3)=O)(CC2)C1 O=C(CCCCCOc1ccccc1)N1CCN(C(C2CCOC(=O)CC2)=O)CC1 CC1=C(C(=O)NCC2CCN(C(c3cn(C)n(C(C)C)c3=O)=O)CC2O)CCO1 c1(NC(C(N2C(CNC(C(C)=O)=O)CCC2)=O)=O)cccc2ccccc12 C(CS(=O)(=O)c1ccc(C(=O)NC2CCCC2N(c2ccccc2)C)cc1)OC C1(NC(Cc2cccc(OC)c2)=O)CN(C(=O)CC(C)C2CC2)C2(CCOCC2)C1 c1(NC(c2csc(S(=O)(=O)N3CCCC3)c2)=O)ccc2c(c1)nc(O)n2C1CC1 CC1OCCCC1C(=O)NCc1ccc(CNC(c2sccc2CO)=O)cc1 C(CN=S(C)(C)=O)NC(CC(C)NC(C1CC(OC)C1)=O)=O CCC(CNC(=O)CC1CC2(C1)CN(C(C1(C(=O)OC)CC1)=O)C2)C(C)(F)F N1(C(Cn2nnc(C)n2)=O)CCC2(CC1)CN(C(=O)C(F)F)C2C(C)C C12(CNC(c3cccc(F)c3Cl)=O)CCCC1CN(C(=O)CC1CC13CC3)C2 C1(C(=O)NCC(C(CC)C)C)CN(C(C2(C)COC2)=O)CC(C)(C)C1 c1(OC2CCOC2)ccc(O)cc1C.C(=O)(COCCOC=O)N(CC)CC.CCN.C c1(OC)cc2cc(c1)NC(=O)N2.C1(C(=O)N(C)C)CCC(F)(F)C1 C(CC1NC(=O)c2ccccc21)OC(c1c(F)ccc(Br)c1Cl)=O Cc1ccnc(C(C)(C)C(=O)NCCCN(C(=O)CC(=O)NCC(F)(F)F)C)c1 C1(CC(=O)N(CCO)CC)CN(C(C2(CC)CCOCC2)=O)CCO1 C12(C(=O)NCC3N(C(c4cc(SC)oc4)=O)CC(OC)C3)CCC(CO)(CC1)C2 N1(C(C=C)=O)CCC(C(=O)NCC2CC(F)(F)C2)C(O)C1 N1(C(c2cn(CCC)nc2)=O)CCCCC2(CCN(C(=O)CSC(F)F)C2)C1 CC1(C(=O)NCCCOCC2C(NC(c3csc(C(F)F)n3)=O)C2)CCCC1 Cc1cncc(C(N2CCC(C(C)(C)C)(CNC(c3snc(O)c3Cl)=O)C2)=O)c1 c1(-c2cc(C(N(C3CC(C(N)=O)C3)C)=O)n[nH]2)ccccc1F C1(CNC(c2cnc(C)s2)=O)CN(C)CCN1C(C1CC2(CC2)CO1)=O C=CCCC(C(=O)NCC(C)N(CC)CC)NC(c1ccccc1CO)=O C12(NC(C=C(CCC)C)=O)CCCC(CN(C(c3cnn(C)c3C(F)F)=O)C1)C2 N1(C(C2(C)N(C)CCC2)=O)CCCC(F)(CNC(C2(C3CCCO3)CC2)=O)C1 Cc1cnnc(O)c1C(N1CCC(C)(CNC(=O)CC2(C)CCOCC2)C1)=O CCCC(CC)C(=O)NCC(O)CCNC(c1cnc(CC(C)(C)C)s1)=O CCC(C)(O)C(=O)NCC(C)C(=O)NCCC12CC(CCO1)C2 N1(C(COCCC=C)=O)CCC(C)C1CNC(c1coc(C)c1)=O N1(C(CC2OCCN(C(C(CC)C(F)(F)F)=O)C2)=O)CCN2C(=O)CCC2C1 C(=O)(C1=NOC2(CCC2)C1)NC(C(C)C)C(=O)NCC(C1CCCC1)C CCC(CC)C(F)C(=O)NC1CCCC1CNC(=O)CCc1ccco1 C(C)(CNC(c1nc(C(F)(F)F)cn1C)=O)(C(C)C)NC(CSCCOC)=O.C(=O)OC c1(C(C)C)csc(C(C)NC(c2nnnn2C2CC(F)(F)C2)C2(CCl)CCC2)n1 Cc1ccc(C(=O)NC2COCCC2NC(c2cnc(C3CC3)nc2)=O)cn1 O=C(N=c1[nH]nc(CC2CC2)s1)N1CCC2CC2C1 c1(C(=O)NCC2N(C(C(C(C)C)NC(N)=O)=O)CC2)cccc(Br)c1N N1(C(C(C)OC)=O)CCC(NC(c2cnn(-c3ccccc3Cl)c2)=O)C1C CON1CC(C(=O)NC2CCCC2C(=O)N(CCCN(C)C)C)CC1=O c1(NC(C2CCC(CNC(c3cncc(Cl)n3)=O)CC2)=O)cc2ccccn2n1 C(C(=O)NCCOCCN(C(=O)Cc1nccs1)C)(C(C)C)SCC CC#CC1CCN(C(=O)C(Cn2cncn2)NC(c2cnn(C(C)C)c2)=O)C1 c1(C(=O)NCCCC2(NC(C3CC=CC3)=O)CC2)cnn(CCO)c1 c1(C(N2C(C)(CNC(CC3(OC)CCC3)=O)CCC2)=O)cc(O)c2ccsc2c1 CC1(CNC(c2ncnc(O)c2F)=O)CCCN(C(C23CCCC2CCC3)=O)C1 C1(C(=O)NC2CCCN(C(c3scc(C(C)=O)c3)=O)C2)CC(=O)NC(=O)N1 C1(C(=O)NC(C(C)(C)NC(C2CCC(CC)O2)=O)C)CC(C)(C)C(C)(C)C1 C12(C(=O)NC3CN(C(CNC=O)=O)CC4(C3)CCC4)CC3CC(C1)CC(F)(C3)C2 C1(OC)CC(NC(=O)CCC=Cc2ccccc2)CN(C(=O)C(C)CO)C1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NCC(CCSC)OCC C1(C(=O)NC2CC(CNC(=O)OC)C2)(CO)CC1(F)F C12(NC(CCCC(=C)C)=O)CCCC1N(C(=O)CN1CCCNC1=O)CCC2 C1(CC)CCCC1NC(c1coc(C2CC2)n1)=O.c12ccc(o1)CNC(=O)CC2 N1(C(C(CCC=C)(C)C)=O)CCC2(CCC2)C(NC(C2CCOCC2(C)C)=O)C1 N1(CCNC(=O)NC(C)C(N2CCCCC2)=O)CCC(C(F)F)CC1 N1(C(c2c(OC)cc(N)cc2)=O)CCC2CCCC12CNC(=O)CN(C)C(C)=O Cc1nn(CC(F)F)c(C)c1C(=O)NCC1C(=O)NCCC1C N1(C(c2ccc(CC)o2)=O)CCCN(CCCCNC(C2CC(=O)N2)=O)CC1 N1(Cc2nccc(CC)c2)CC2CCC1CN2C(=O)NCc1cc(C)ccc1F CN1CCCC(CCNC(C2CCC2CNC(=O)Cc2cn[nH]c2)=O)C1 CC1(NC(c2cc(O)ncn2)=O)CCCN(C(=O)C=Cc2ccccc2)C1 c1(C(=O)NCC(C)N(C(=O)CCCN2CCCC2)C)cccc2c1ncn2C CC1(C)CCC(C)(C(N2CCC(O)(CCNC(=O)C#CC3CCCC3)C2)=O)CC1 c1(C(N2CCC(CC=C)(NC(=O)C=CCF)CC2)=O)cc(Cl)cc(F)c1F N1(C(c2c(OC)cc(Cl)cc2)=O)CCC(NC(=O)CN2CCOCC2)C(C)(C)C1 CCC(C(=O)N1CC2CC1CN(C(C1(SC)CCC1)=O)C2)C(C)(F)F C1(NC(CCOCC#C)=O)CCN(C(C2CC(OCC)C2)=O)C12CCC2 C(=O)(C(C(C)C)SN(CC)CC)NCC(CCC)N(C)C.C1(=O)C(C)N1 S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(CO)s1)NCC(CC)N1CCCC1 CC(C)C(C(=O)N1CCC2CN(C(c3ccnn3CCF)=O)CC12)C(C)C C1(C)(CC)C=C(C(=O)NCCCCC(CO)NC(=O)CCc2c(C)noc2C)C1 N1(CCc2cn(CC)nc2)CCOC(C)(CNC(C2(C)CCNC2=O)=O)C1 c1(C(=O)NC(C)CCCNC(C2CCC(F)C2)=O)cnc2nccn2c1 C1(NC(c2ccc(CNC(C)=O)s2)=O)CCC(C)N(C(=O)C(O)C(F)(F)F)C1 c1(NC(C)=O)cccc(S(=O)(=O)NCC23COCC2C3)c1 n1(C(C(=O)OC)C)cc(CNC(C2CC2C(C)(F)F)=O)nn1 CP(C)(=O)c1ccnc(-c2nc(-c3ccccn3)nn2CC2CCCO2)c1 N1(C(c2cc(C)c(O)nn2)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC(C)C1 C(CN=c1cc(C)c(S(=O)(=O)N2CCC(S(C)(=O)=O)CC2)c[nH]1)OCCOCC C#CC1(C(=O)NCCOCC)CCN(C(C2CC(CCO)C2)=O)C1.C(CCC)N c1(OC(C)C)cc(C(=O)NCC2CC(NC(=O)CC3CC3(C)C)CC2O)ccn1 C(=O)(C(O)CC(N)=O)NC(CNC(C=C(CCC)CCC)=O)(C)C1CCC1 CCC(CC)C(F)C(=O)N1CC(O)(C(C)NC(C2CC2C2CCCO2)=O)C1 O=C(CS(=O)(=O)Cc1cccs1)NCC12CC1CN(C(C1C3(CC3)C13CC3)=O)C2 C1(CNC(C2CC2CF)=O)CN(C(=O)COCc2ccccc2Cl)CCO1 N1(C(C2N(C)CC2)=O)CCC(O)(CCNC(=O)CC2CSC2)CC1 c1(C(=O)OCC2CC(NCC)C2)cc(F)ccc1CC C1(C#N)(C(=O)NC2CC3(C(C(N4C(C)CCCC4)=O)C3)C2)CCOCC1 C1(NC(C(C)OCC=C)=O)COCCN(C(c2cn(CCOCC)nc2C)=O)C1 Cc1ccc(-c2cc(C(=O)NC(CNC(c3occc3C)=O)CO)no2)c(C)c1 c1(C(=O)NC2C(C(=O)Nc3c(C(=O)OC)n[nH]c3)C2)cc(C)c2cc[nH]c2c1 n1(CCOC)c(C(N2CC3C(C2)C2(OC)CCC(C2)O3)=O)cnc1O.C(=O)O.OC C(C1CN(C(=O)CC2C=CCC2)Cc2ccccc21)NC(c1scc(OC)c1)=O CC1CCOC1C(=O)NCC1(CNC(c2cc(C3CC3)ns2)=O)CC1 C1(CC)CN(C(c2ccncc2Cl)=O)CC1C(=O)Nc1conc1C C1(C(=O)NC(C2CC(F)(F)C2)C#C)CCCN(C(=O)CCC#CC)CC1 C1(F)(CNC(CC2CC(NC(C(C)SC(F)(F)F)=O)C2)=O)CCOC1 C1(CC)COC(C)(C)CN1C(C1CC2CCC(C1)N2C(=O)CC(C)(C)C)=O N1(C(=O)Cn2ncnn2)CCN(C(C2CCC3(CCC3)O2)=O)C(CCO)C1 C=CCCCCCC(=O)NCCN(C)C(C1(COC)CC(=C)C1)=O c1(CN2C(C(=O)Nc3c(OCC)nccc3)CCCC2)ccn2cncc2c1 c1(COC)cc[nH]c1C(=O)NC1CCC1C(=O)NC1(CCF)CC(O)C1 C1(N(C(COCCC(N2CC(O)(CC=C)C2)=O)=O)C)CC12CCOC2 C(=O)(C1CC(Nc2ccc(OC)c(C(C)=O)c2F)c2ccccc21)OCC CC1OC(C)CC1NC(C1(NC(=O)C(=O)NCC(F)F)CSC1)=O C12CN(CCC13CCOCC3)C(=O)CCNC2.C1(CC(=O)NC2CC2)CC1(Cl)Cl N(C(=NCCc1ncccc1C)NCC1C=CCC1)C(C=C)C CCC(C(=O)NCC1(C)CN(C(c2ccnn2CC)=O)CC1C)C(C)(F)F c1(C(=O)NCC2N(C(CSCC#C)=O)CCCC2C)ccc2c(c1)CCC(=O)N2 c1(-c2nnc(CCCCC)o2)ncccc1OC.C(C)C c1(N(CN2CCN(C(C)NC(=O)OC)C2=O)C)ccc(F)cc1F N1(C(C(CCC)=O)=O)CCC(F)(C(=O)NC2(c3noc(C)n3)CC2)CC1 c12cccc3c1OC(C3)C(=O)OC2.c1(C(=O)OC)ccc(OC)c(OC)c1 C1(CCOC)(NC(C2(Cl)CC23CCC3)=O)CCN(C(=O)CN(C)C2CC2)C1 Cc1oc(Cl)nc1C(=O)NC1CC(CNC(c2cncc(OC(C)C)c2)=O)C1 Cc1cccc2nc(C(=O)NC3CCCN(C(C45CC(CO4)C5)=O)CC3)cn12 N1(C(C2CCCN(C(c3cc[nH]n3)=O)C2)=O)CCCCC(F)(F)C1 CCCCC(CCCC)C(=O)N1CCC(CNC(=O)C=CS(C)=O)C1 C1(NC(CN(C)C2CC2)=O)CN(C(C2(N(C)C)CCCSC2)=O)CC2(CCC2)C1 C=CC(C)(C)C(=O)N1CC2CC1C2NC(=O)CNC(c1ccoc1)=O C(=O)(C1=NNC(=O)CC1)N1CCC(C)C(CN=c2[nH]nc(-c3ccccc3)o2)C1 N1(C(CCc2n(C)ccn2)=O)Cc2[nH]nc(C(N3CCOC4CC34)=O)c2C1 C(=O)(CC(CN(C)C)CC)NCC(CC(=O)N1C(CC)CC1)OC C(CNC(=O)CSCc1ccccc1Cl)(CC(C)C)NC(C1C(C)(CC)C1)=O N1(C(c2c(CC)n[nH]c2)=O)CCCCC(CNC(C2CC2c2ccn(C)n2)=O)C1 C(c1c(F)cccc1F)=CC(=O)NC1CC(NC(=O)CC2(O)CC2)C12CCC2 C(=O)(C1SCc2cccnc21)NC12C(CN(C(C(C)=CC)=O)C1)COCC2 Nc1cc(F)c(F)cc1C(=O)NCC1CCCN(C(c2cccnn2)=O)C1 C1(c2c(OC)cccc2)CCN(c2nc(C(F)F)ns2)CCO1 C1(N(C)C(C2(S(C)(=O)=O)CC2)=O)CN(C(=O)C(c2cccn2C)=O)CC1(C)C C(=O)(C#CC(C)(C)O)NC(C1CCN(C(C(C=CCCC)O)=O)C1)(C)C c1(SCC(C2CN(C(C3(NC(c4cc[nH]c4)=O)CCC3)=O)C2)=O)ccccc1 c1(C(=O)NC(C)CCNC(C2CCC2CF)=O)ccc2c(c1)COCCN2 CC1CN(C(=O)CCC2(C(=O)C(O)c3ccsc3)CCCC2)CCO1 C(=O)(C(O)CC(C)(C)C)NCC(C(C)(C)C)NC(c1cnccc1C#N)=O N1(C(=O)Cc2ccc(Cl)cn2)CC(NC(C2(CO)CCOCC2)=O)CC(F)C1 c1(NC(C2OCCC(NC(CC(C)C)=O)C2)=O)ccc(F)c(CN(C)C)c1 c1(N2CC(NC(c3ccc(CC)c(F)c3)=O)C(C)C2)ncn(C)c(=O)c1Br CC1CC(NC(C2(NC(=O)CC3CC(F)(F)C3)CSC2)=O)CCS1 C(C)(C)(CC(=O)NC(c1ncn(C)n1)C)NC(C(CC)N(C)C)=O C(=O)(CCC(=O)N1CC(NC(c2sccc2-n2ccnn2)=O)C(COC)C1)NC N1(C(C(CC(C)C)Cn2cc(CCC(=O)CCO)nn2)=O)CCC(=C(Br)Br)CC1 CC1(CNC(C2(C)CC2(F)F)=O)CN(C(C2CCC(F)(F)CC2)=O)CCO1 Cc1ccc(C(=O)NCC2CCCCN(C(c3c(C)noc3C)=O)C2)c(Cl)c1C CC(C)C(C)(O)C(=O)NCC(=O)OCc1ccc(Br)cc1F C1(C(C)NC(c2cn(CCO)nn2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 C1(C(N2CC3C(CNC(CNC(=O)OCC)=O)C3C2)=O)CCC(=C(F)F)CC1 c1(NC(c2cc(Br)cnc2Cl)=O)ccc2c(C(F)(F)F)cccc2n1 Cc1cc2c(C(=O)N(C(C)CNC(c3cc[nH]c4nccc3-4)=O)C)nccn2n1 c1(OC)ncc(C(=O)NC2CCN(c3ncnc(Cl)c3C)CC2C)c(C)n1 N1(C(CCn2cc(CCOC(C)=O)nn2)=O)CCC(O)(C(c2ccco2)C(C)C)C1 N1(C2CCCN(C)C2=O)CCC(F)(F)C(CNC(c2ccns2)=O)C1 C(=O)(C1=C(N)CCC1)OCCCN1CCCC(C)C1 c1(CNC(C2(C)CC2C(=O)Oc2ccc(F)cc2)=O)ccc(F)c(C#N)c1 C1(NC(c2cc(SC)oc2)=O)CN(C(=O)CC2CCCC23CC3)CC1(C)C Cc1nc(-c2ccc(Cl)cc2)oc1C(=O)NCc1cn(C2CCCC2(F)F)nn1 CCC(C(=O)NCC1CCCN(C(=O)C(C)SC)C1)C(C)(F)F c1(C(=O)NC2CN(C(C=C(C)Cl)=O)CC2C2CC2)cn2cccc(C)c2n1 c1(C(N2C(CCNC(C3CC(=O)NC3)=O)CSCC2)=O)cc[nH]c2nccc1-2 N#Cc1cccc(C(=O)NC2CN(C(c3cncc(Cl)c3)=O)CCC2(F)F)c1Cl C1(C(=O)NCC(c2cn(C)nc2)O)CC2(CCC2)CN1C(C1CC(C)(C)C1)=O C=CC(C)(CCOC)C(=O)N1CC(NC(=O)CCC=CBr)C(F)C1 Cc1nn(C)c2sc(C(N3CCC(C4(NC(c5nncn5C)=O)CC4)C3)=O)cc12 N1(C(c2c(C(C)C)ocn2)=O)CC2CC(C(N3CCC3c3ccco3)=O)(C2)C1 C(c1cccc(Cl)c1)=C(C(=O)N(CC(CC)NC(C1(C#N)CCCOC1)=O)C)C c1(C(N2CC(CNC(CCOCC)=O)C(C)(C)C2)=O)ccc2c(Cl)nccc2c1 C1(C(=O)NCC2(NC(c3c(N)cn(C)n3)=O)CCCCC2)CC(=O)NC1(C)C Cc1cn2nnc(C(N3CCN(C(C4COC(C)C4)=O)C(C)C3)=O)c2c(O)n1 c1(C(N(CC)CC2CCCN2C(C2CC2F)=O)=O)ccc(C)nc1OC N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(NC(=O)Cc2cncs2)CC(F)C1 c1(OCC)ccc(C(N2CCN(C(=O)C#CC(C)C)CC2CO)=O)c(Cl)c1 c1(NC(C2(C)CNC2)=O)ccccc1CC1CCS(=O)(=O)C1 N1(C(c2cnc(CC)[nH]2)=O)CCC(C(C(C)C)NC(c2ccc(Cl)cn2)=O)CC1 c1(CC)ccc(CN2CC(C(=O)NCC3CCCC3C)(CC)C2)cc1C c1(C(C(=O)OCC2C(C(=O)O)C2)(F)F)ncccc1F C=CCC(C(=O)NCC1(F)CC(NC(=O)C(c2ccccc2)=O)C1)NC(C)=O C=CCC(C)(C)C(=O)NCC1CCCCN(C(=O)C(CC=C)NC(C)=O)C1 n1(CC)cnc2[nH]c(=NC(C)c3cnn[nH]3)nc(N3CCC(F)(CO)CC3)c12 C1(OC)CC(C(=O)O)CN(C(C2CC2(C)C)=O)C1 N1(C(c2cc(C)nc(C)c2)=O)CC(NC(c2[nH]cc3c2CCC3)=O)CCC(O)C1 C1(C)(CNC(C(CN(C(CC2CC(=C)C2)=O)C)C)=O)CCCC(=O)N1 c1(C(C)C)nocc1CNC(=O)C(C1CCOC1)NC(=O)CC(=O)N(C)C N1(C(c2cc(OC)c(C)cc2)=O)CC2CCCC(NC(C3CCCC3C)=O)C2C1 C1(=O)CCN(C)CCN1C.C(CCOC)NC(C1C(C(=O)NC)C1)=O c1(C(N2CC=CC(NC(C3C(C)(C)CC3)=O)C2)=O)ccc(C#N)c(O)c1 c1(C(N2C(CNC(c3c(C)coc3C)=O)C(C)(C)CC2)=O)cc([N+](=O)[O-])nn1C c1(NC2(CC=C)CN(C(C3(C(F)F)CCCO3)=O)C2)ncnc2ccc(O)cc12 c1(CC(N)CN(C(=O)Cc2cocn2)C2CC2)ccc(Cl)cc1 N1(C(C(CC)O)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)NC(=O)OC(C)(C)C)C2 C12(NC(Cc3nc(C)sc3)=O)CCN(C(=O)CCCNC(=O)C3CC3)CC1C2 c1(C(N2CCOCC2CCC)C(=O)NCC=C)ccc(C)c(C)c1 c1(C(=O)NC2CCN(C(c3nc(C)oc3C)=O)CC2)cnc2ccccn12 N1(C(C2(COC)CCC2)=O)CCC(C)C(CNC(c2ccc(O)cc2C)=O)C1 c1(C(=O)NCC(CC)(CC)NC(=O)C(C(C)C)C(C)C)ccn2cc(C)nc2c1 c1(C(N(CCCNC(C2(c3cccs3)CCCC2)=O)C(C)C)=O)cnc(N)cn1 N1(C(C)=O)CCOC(CNC(=O)CCc2ccncn2)C1.N12CCC1C2=O Cc1ccc2cccnc2c1C(=O)NCCCC(C)(C)NC(=O)C(C)(F)F Cc1cnn(C(C)C)c1C(=O)NCC1(CN(C)C(C2CC2Cl)=O)CC1 C1(O)(CNC(C2(CC=C)CC2)=O)CC(C(=O)NCC(CO)N(C)C)C1 C1(CN(C(CCOCCC)C)C)CN(C(=O)CC2CCCC(=O)C2)CC1CCC c1(C(=O)NCCCCNC(=O)C2CC2)ccc(-c2cccs2)cc1F c1(C(=O)NCCC(C)NC(C2(C(F)(F)F)CCCC2)=O)c[nH]nc1-n1cnnn1 N1(C(C(C)=O)=O)CC(C2CCCCN(C(c3cn(-c4ccccc4)nn3)=O)C2)C1 C(C)(C(=O)N(CC(=O)N(C12CC(C1)C2)C)C1CC1)[SH](CCCC)C1CC1 Cc1cc(C(N2CC(F)(F)CC2CNC(c2n[nH]c(O)n2)=O)=O)ccc1F C1(CN(C(C(C)N2CCC2)=O)C)CN(C(c2cnc(Cl)cc2N)=O)CCO1 c1(C(N2CCN(CCN(C)C(C3(Cl)CC3)=O)CC2)=O)ccn2cnnc2c1 C(C(=O)NCCC(=O)O)(C(C)(C)C)n1cc(-c2cccc(C(=O)OC)n2)nn1 C=CC1OCCCC1C(=O)NCC=CCNC(=O)CN1CCCNC1=O c1(NCC(C2CCC2)NC(CN(CC)CC)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(C(C)N=[N+]=[N-])=O)CC=C(C(=O)N(C2CCCCCCC2)C)CC1 c1(C(N2CCCCC2CCO)=O)cc2cc(-c3ccsc3CO)cnc2[nH]1 C1(CC)CCOC1C(N1CC(C(=O)NCCC2CCCS2)(CC)C1)=O N1(C(COCC(=C)C)=O)CCC(CN(C(=O)C(C)n2cccc2)C)CC1 C1(C(=O)NC(CC=C)C2CC2)CCCC1CNC(C1C=C(C)CS1)=O c1(SC)cc(=NC(=O)C23CC(NC(c4cnn5c4OCC5)=O)(C2)C3)[nH]n1C c1(C(=O)NCC(CNC(c2cc(C(F)F)ncn2)=O)OC)c(Cl)nsc1Cl C=C(CNC(C1CCN(C(C2CC2COCC)=O)C(C)C1)=O)c1ccccc1 c1(OC)ccc(F)c(C(N2CCC(N(C)C(c3ccc(F)c(C)c3)=O)C2)=O)c1F c1(CCNC(C2C(CNC(=O)CN3CC=CC3)CCO2)=O)ccncc1 c1(C(N2CC(C(N3CCCC3)=O)C(O)CC2)=O)nc2ncccn2n1 c1(OCC=CC(=O)NCc2ccc(OCC)cc2)cccc(Cl)c1Cl C1(C(N2CCC(O)(CO)CC2)=O)CC(F)(F)CN1C(C1CC(F)(F)C1)=O c1(NCC(=O)NC(C(=O)OCC)CCC2CC2)ccc(C#N)c(OCC)c1 C(=O)(C1=CCCCO1)N(CCNC(=O)C(C)(C)C1CCOCC1)CC C(C(O)CC(=O)Nc1cncc(N(C)C)c1)NC(CC(C)O)=O C1(F)(CF)CCCN(CN)C1.c1(CCC(=O)C(CC2CN(C(C)=O)C2)=O)nccn1C CCCCCCC(C)C(=O)NC(CCC(C)C)C(=O)NCC(C)(C)C(C)(F)F Cc1noc(C(N2CC(N(C)C(C3COCC3(C)C)=O)C2)=O)c1C(F)(F)F c1(C(N(CCOCCCNC(Cc2cc(C)no2)=O)C)=O)n[nH]c2c1NCCC2 CC1(C)C(C(=O)NCCC2(NC(=O)C=CC3CCCC3)CC2)C1c1nc[nH]n1 C1(C2(O)CCN(C(c3ccc4ncnn4c3)=O)CC2)(NC(C2C(=C)C2)=O)CC1 C1(C(=O)NCC(CO)NC(c2[nH]nnc2C2CC2)=O)C2CC3CC(C2)CC1C3.OC CCS(=O)(=O)c1ccccc1C(N1CC(CNC(=O)C(C)CSC(F)(F)F)C1)=O c1(OC)cn(CC(N2CCCC2CNC(C2CCC(=O)N2C)=O)=O)c(C)cc1=O c1(C(CN2CC3C(CNC(C(C=C=C)C)=O)C3C2)=O)c(F)ccc(Cl)c1F C12(CNC(CCCC)=O)CCCCC1CN(C(c1coc(CC)n1)=O)C2 C1(NC(C2CCC(N(C(COC(C)=O)=O)C)CC2)=O)CCCC(C)CC1 CC1(C(N2CCC(CCCNC(C3(C4CC4)CC3)=O)CC2)=O)CC(F)(F)C1 c1(C(=O)NCC2(N(C(C(CC)OCC)=O)C)CC2)n[nH]c2c1CCC2 N1(C(CC(CC)OC)=O)CCCC2(NC(=O)CCc3cc(C)no3)CC2C1 C(=O)(C(C(=O)NCCCC(C)(C)NC(C1CCC(C)(O)CC1)=O)C(C)C)OCC c1(CC)nnc(CC(N2CC(C(=O)NCc3cccnc3)C2)=O)o1 C1(NC(c2cnc(C)s2)=O)CCN(C(C23CC(C2)C(C)O3)=O)CC1F c1(OC(C)C)ccc(C(F)CNC2CCN(S(C)(=O)=O)CC2)cc1 N1(Cc2c[nH]c3ccc(OC)cc32)CCc2cc(NC(=O)C(Cl)(Cl)Cl)ccc2C1 C1(NC(=O)NCCCSC)(CNC2CCCCN2c2ccncn2)CCN(C)C1 N1(CC)CCCC1C(=O)NCC1CC(NC(c2coc(C(C)(C)C)n2)=O)C1 CCCC(CCC)C(=O)N1CCC(C(=O)NCC(O)C(C)(C)O)CC1CC C1(C(N2CC(C(C)NC(c3cc(C(F)F)[nH]n3)=O)C2)=O)CCOC(C(F)(F)F)C1 CC1=NN(C)C(=O)C1CC(=O)NC(C)CNC(=O)Cc1ccsc1C c1(NC(c2cc(-c3ccc(C4(O)CCC4)cc3)cnc2F)=O)ccc(F)cc1Br c1(C(=O)NC2CC(CNC(=O)C(c3ccc(F)cc3)O)C2)cccc2c1CCO2 c1(NC(c2n(C(CC)(C)C)nnn2)(C)CC2C=CCC2)cccc(CCO)c1 CCCC(C)(CC)C(=O)NCC1CN(C(=O)C(C)(C)CC)CC1(F)F C1(O)(CCNC(=O)C(c2ccc(Cl)cc2)O)CCN(C(=O)CC2CC=CC2)CC1 CCC(C)C(O)C(=O)NCC1COC(CNC(c2cc(O)ccc2F)=O)C1 CC1(C)CCCN(C(=O)COCC2CCC2)C1CNC(C1CC2OC1C1CC21)=O C(CN=C(NCC1CCCO1)N(C)CC1(O)CCC12CCC2)OCC c1(C(=O)NCCCNC(C23COCC2C3)=O)ccc(=O)n2c1CCC2 n1(CC(N2CC(CNC(c3coc(Cl)n3)=O)OCC2)=O)cnc2ccccc12 N1(C(c2n(CC)ncn2)=O)CC2CC1CN(C(=O)C=CC1CCCO1)C2 C(=O)(C(C(C)NC(=O)CC1=CCCC1)C(C)C)Nc1c(C)nc(Cl)nc1 Cc1nc2n(n1)CC(C(=O)NCCCNC(C1CCC3(CCC3)OC1)=O)CC2 C#CCCCCCC(=O)N1CCC(C2CCCN2C(=O)C=Cc2cccn2C)C1 C1(CNC(=O)CN2CCC2)CCCN(C(C2C(F)(F)C23CCC3)=O)CC1 c1(SC)ccc(O)c(C(N2CCC(N(C(=O)C(C)P(C)(C)=O)CC3CC3)C2)=O)c1 N1(C(c2csc(CC3CCCC3)c2)C(=O)NCCCC)CCC(C)CC(C)C1 C1(CCOC)CN(C(=O)C(C)CC)CCN1C(c1cc(C(N)=O)c[nH]1)=O n1(CC(N2CCC(N(C(C(C)OCC#C)=O)C)C2)=O)ccc(O)nc1=O N1(C(C(c2ccccc2O)OC)=O)CCN(C(c2ccnn2C(F)F)=O)CC1 c1(NC(=O)NCC(=O)NCC2(O)CN(C(C3C(CC)C3)=O)C2)c(F)cccc1F C1(C(=O)NCCC(C)CCNC(=O)CCN2CCOCC2)CN(C)C(=O)CCO1 C#Cc1cnn(CC(=O)NC2(CCCC(=O)NCC(C)(C)N(C)CC)CCC2)c1 c1(C(C)C(=O)NCCN(C(c2cnc[nH]2)=O)CC2CC2)ccc(Cl)cc1 CC(=Cn1ccnn1)C(=O)N1CCCN(C(c2c(C)nc(C)nc2C)=O)CC1C C1(CNC(c2nc(C#C)sc2)=O)CC2(CC2)CN1C(=O)Cc1ccc(Cl)c(Cl)c1 C1(C(N2CC3CCC(C(=O)NC)CC23)=O)C2C3CC4C1C1C2CC3C41 C1(NC(C=CC(=O)N(C)C)=O)CCCCC1C(N1CCC(CO)(CF)C1)=O C(C)(C)(C(=O)NCc1cc(C(N2CC(n3cnnn3)C2)=O)n[nH]1)NC(C)=O C(CC(N)CC(C)(C)C)N.C(CCC)CCC c1(CCCC)n[nH]c(=NCc2cnn(C3CC3)c2)s1 C=CC(C)(CC)C(=O)N1CC(NC(c2csc(Br)c2C)=O)C(C)(C)C1 Cc1ccn2cc(C(N3CCC(N(C(=O)CC4CC4C4CC4)C)C3)=O)nc2c1C c1(C(N(C2CCCN(C(C3ON=C(CC)C3)=O)CC2)C)=O)c([N+](=O)[O-])cnn1C C=CC1(NC(=O)C(C)(C2CCC2)NC(c2ccon2)=O)CCCC1 C1(NC(C(C)=CC2CC2)=O)CC2CCC1N(C(c1ccccc1CO)=O)C2 c1(C(N2CCCC(NC(CC(=O)OC)=O)C2)=O)cc([N+](=O)[O-])sn1.C1(C)CC1 C1(CC(=O)NC)(CN(C)CC2CCN(C(c3ccc(C)o3)=O)C2)CCCCC1 CC1CN(C(c2snc(Cl)c2Cl)=O)CC(C)N(C(c2cccn3ncnc23)=O)C1 n1(CC(=O)N(CCC(C)N(C(C2(N(C)C)CC2)=O)C)C)nnnc1C1CC1 C1(C(=O)OC(C)(C)C)(CC)CCCCN1C(C1C(C)C1(C)C)=O N1(C(CC(C)(F)F)=O)CCCC2(C1)CN(C(c1c(Cl)cnn1C)=O)CCO2 C1(CNC(c2c(CC)nccc2)=O)CCN(C(=O)CCOC(C)C)CC1C C1(C(=O)NCC(C)CNC(C2CC(=C3CCC3)C2)=O)OCC1(C)C C1(NC(C(C)(C)C2CC2)=O)CCN(C(C2CCOC2)=O)CCC1CO c1(C(N(CCNC(C2CC(C(=O)OC)C2)=O)C2CC2)=O)nc(C)ccc1F N1(C(COCC=C)=O)CCOCC(NC(=O)C=C(CC)CC)C1 N1(C(C(C2CC2)OC)=O)CC2(CCC2)CC1C(N1CC(C)(OC(C)C)C1)=O C1(F)(CNC(C2CCS(=O)CC2)=O)CC2CCC(C1)N2C(C1CC2CCC1O2)=O CC1(C)CC(NC(=O)Cc2c(F)cccc2F)CN1C(=O)CCc1nccs1 C(=O)(C(CO)C(F)(F)F)NCC1CC(NC(c2cccc(OC)c2C)=O)C1 C(=O)(C1=CC2(CCOCC2)C1)N1CCC(C)NCC1.c1ccc(C(N)=O)cc1 C(=O)(NNc1cc(Br)c(F)cc1F)c1cncc(CN(C)C)c1 C1(N(C(C)(C)C)C(=O)OC)CC2(CNC2)C1.N1(C(C(C)O)=O)CCC(NCC#N)C1 Cc1ccnc(C(=O)N(C2CN(C(c3ncoc3C3CCCC3)=O)C2)C)n1 S(=O)(=O)(c1cc(C(=O)N=c2cccn[nH]2)n(C)c1)NC(C)C(=O)N1CCCC1 CC1CN(C(C2(C)CCCS2)=O)CC1CCNc1cc(O)ncn1 C1(NC(c2c(OC)c(C)cs2)=O)CCN(C(C2CC3(CC3)CO2)=O)CC1(C)C N1(C(CC(C)F)=O)CC2(CCCC2NC(=O)CN2CCNC(=O)C2)C1 C1(CC)CC(=O)N(C(C)OCCC(=O)NC2CC(CNC(=O)C(=O)NOC)C2)C1 C(=O)(C(F)C(=O)NCC(C(=O)N1CC(OCC(F)F)C1)N(C)C)OCC C(=O)(C1=CCC(C)CC1)N(CC(=O)Nc1c(C)c(O)ccc1)C C1(CC)CN(C(=O)CC2CCSC2)CCC1NC(C1CC(O)C1)=O C1(C(N2CCC(O)(c3cn(-c4ccc(O)nc4)nn3)CC2)=O)CC12CCCCC2 c1(C(=O)NCC2N(C(c3cnc(CC)[nH]3)=O)CC2)cnn2ccc(Cl)c(F)c12 CC(=O)CCCCCCC(=O)NC1CC(C)N(C(c2cnoc2C)=O)C1 C(=O)(C(CC(N)=O)NC(=O)C(C)OCC(C)C)NC1(CCC)CCC1 C(=O)(C(C)(C)CC(F)(F)F)N1CCCC(CNC(C2C(CCC)CCC2)=O)C1 c1(CC)nn[nH]c1C(=O)NC(C1CCCN1C(=O)C(C)SC)(C)C CC1CCN(C(C23CC(CO2)C3)=O)C1CNC(=O)CCc1cncs1 N1(C(c2ccc(CO)o2)=O)CCCC2CN(Cc3cccc(O)c3)CCC12 CC1=C(C)CC(C(=O)NC2(CNC(c3c(Cl)c(C)nn3C)=O)CCCC2)CC1 c1(C(=O)NCCOCCN(C)C)csc(C(=O)Nc2ccc(Br)o2)n1 C1(C)(CCC(=O)N(CCC(C)NC(=O)CCCn2cncn2)C2CC2)CC1(F)F C(C)(C(CC(=O)NCC1(CCOC)CC1)NC(=O)CN=[N+]=[N-])OC c1(NC)cnccc1C(=O)NCCO.N12CCCC(C1)c1cn(nn1)CC2 C1(C(N2CCC(C)(CCO)C2)=O)CC2(CC2)CN1C(c1cnn2c1OCC2)=O N1(C(C=CC)=O)CCC(O)CC1C(=O)N(CC(c1ccccc1)O)CC(C)C C=CCCC(CC(C)C)C(=O)N1C2CCC1CN(C(c1coc(C(C)C)n1)=O)C2 N1(C(C(CC(=C)C)C)=O)CCC(C)(C)C(NC(=O)COCCCF)C1 C(C)(N=c1[nH]c2c(c(=NC3CCCn4c(O)nnc43)[nH]1)CSC2)c1ccc(C)cn1 N1(C(C=CC)=O)CCC2(NC(=O)CCOc3ccc(F)c(F)c3)CC2C1 C12(C(N3CC(O)(CN(C(c4c(C)nccn4)=O)C)C3)=O)CC3CC(C(=O)N1)C2C3 C1(CC(N2C(C(C)C)COCC2)=O)CN(C(=O)Cc2cnoc2)C(C)(C)C1 CC(C)CC(CN(C)C)NC(=O)C1CC1.c12cc(on1)CCC(=O)N2 N1(C(=O)C=CCO)CC2CCC1C1CN(C(C3(CF)COC3)=O)CC21 C1(NC(c2nccc3[nH]ccc23)=O)COC2(C1)CN(C(C1CCCS1(=O)=O)=O)C2 c1(CC(=O)NC(C)C(CO)NC(C2(C(F)(F)F)CC2)=O)cccc2c1CCC2 N1(C(C(C)NC(CC)=O)=O)CC(NC(c2cc(C(=O)OC)co2)=O)C2(CC2)C1 Cc1cc(C(N2CCCC(O)(CNC(c3cc(C4CC4)[nH]n3)=O)C2)=O)nc(C)n1 N1(Cc2c(OC)nccc2)CC2CC(NC(=O)Nc3cc(CC4CC4)ncn3)C1C2 CC(CCC(=O)NCc1cccc(C(=O)NCCCC2CCC2)c1)S(C)(=O)=O CCCCC(=O)C(=O)NC(C)(C(=O)NCCCn1ccnc1C)C1CCC1 N1(C(C(C)C2CCOC2)C(=O)NCc2ccco2)CCCOCC12CCC2 C1(NC(c2ccc(SC)o2)=O)CC2CCC1CN2C(=O)CN(C)C1CC1 C=CCCC(C)NC(C1(CNC(c2cnc(OC)s2)=O)CC=CC1)=O c1(OC)ncnc(N2CCN(C(=O)Nc3cc(F)ccc3C)CC2CC#N)c1C O=C1CCC(C(=O)NCCOC2CCN(C(c3cc(C4CC4)on3)=O)C2)C1 C(=O)(C(F)C(=O)NC(Cn1cccn1)C(=O)NCC1CCOCC1)OCC N1(C(C(N2C(CC)CCC2)=O)=O)CCCCC(CNC(=O)CCn2ccnn2)C1 N1(CC(=O)CCSCC)CC(OC(=O)C)CC1=O.N1(CC2(C(C)(C)O)CC2)CCCC1 CC(C(C)(F)F)NC(C1C=CCN1C(=O)CSC(C)(C)C)=O N1(C(c2c(OC)scc2)=O)CCCC2(CC(NC(=O)CNC(=O)C3CC3)CO2)C1 c1(C(=O)NCC2(C)C(C)CN(C(=O)CCOC3COC3)C2)cc2ncccc2[nH]1 Cc1[nH]nc2ncc(C(=O)NC(CNC(c3cncn3C)=O)CC(F)(F)F)cc12 C1(N(C(C2C(CCOC)C2)=O)C)CCCCC1N(C)C(c1nn[nH]c1Cl)=O C#Cc1ccc(C(=O)NCc2ccc(C(=O)N(C3CCCC3)CCF)o2)o1 CN1CCCC(CC(=O)NCCC2CCN(C(=O)COc3cnn(C)c3)CC2)C1 Fc1ccc2nc(-c3ccc(-c4nccn4C4CCNC4)cc3)[nH]c2c1 N1(c2c(C#N)ccc(Cl)n2)CCC2CCN(C(=O)CCS(N)(=O)=O)CC2C1 N1(C(CC(C)CNC(=O)C=CC(C)(C)C)=O)CCOC2COCC2C1 CN1CCN(C(C2CC=CCC2NC(=O)CCN2CCOC2=O)=O)CC1C1CC1 C(=O)(C(O)CC(F)(F)F)NCc1ccc(C(N(C)CC2CC(F)C2)=O)cn1 C1(CNC(C(C)(C)SCC)=O)CN(C(c2cnc(OC)s2)=O)CC1C(F)(F)F c1(CC)ccc(C(=O)NCCCN(C(=O)C(F)(F)C(C)O)CC)c(Cl)c1 c1(C(=O)NCCCN(C(C)C)C(C2CCS(=O)CC2)=O)n[nH]c2c1COCC2 CCC(CC(=O)NCCCCCN(C)C(c1cc(C)n(C2CC2)n1)=O)C1CC1 C1(C(=O)NC(CC)CNC(=O)C(C)CF)CCc2ncnc(C)c2C1 c1(N(CCNCC)CC)nc(C(c2nc(OCCOC)n[nH]2)C)cc(C)n1.C1CO1 c1(OC)ccc(C(=O)NC2CC(F)(CNC(=O)C(C)CS(C)=O)C2)c(F)c1F c1(C(N2C(C(C)NC(C(C)C3CC3)=O)CCC2)=O)coc2c1C(=O)CCC2 c1(OC)cc(C(N2CCCCC2CF)C(=O)NCc2cccs2)cc(OC)n1 CC(C)C(C)CC(=O)N1CCN(C(c2ccc(N)c(N)c2)=O)C(CCO)C1 CC(F)(F)C(F)C(=O)N1CC(CC(=O)NC2(C(N)=O)CC2)CC1(C)C CNS(=O)(=O)N1CCC(C(=O)NCCOCCN(C(=O)C(C)N2CCC2)C)CC1 C1(C#N)(C(=O)NCC(C)CNC(c2ccc(CO)s2)=O)CCCOC1 C1(NC(c2sc(C)c(C)c2C)=O)COC2(CCN(C(=O)CN(C)C3CC3)C2)C1 N1(C(c2c(C)cc(C)[nH]2)=O)CC2CCC1CN2C(C1CC1c1cccs1)=O c1(OC)ccc2nc(C(N3CCC3CNC(C34CCC(CC3)CC4)=O)=O)cn2n1 C=C(C)c1cccc(NC(=O)C(=O)NCc2cc(C(C)C)nn2C)c1 C#CC1(C(=O)NC2CN(C(=O)C(C)(C3CCOCC3)OC)CC2C)CCCC1 c1(C(=O)NC(C(C)C)CCN(C)C(c2nsnc2O)=O)scc2c1OCCO2 N1(CCOC(c2ccccn2)=O)CCC(OCc2ncc(CO)o2)CC1 C1(NS(=O)(=O)Cc2csc(-c3ccccc3)n2)CC2(CCC2)C12CCC2 c1(NC(CC2ON=C(CC)C2)=O)ccc(NC(C2CC(=O)CCO2)=O)c(C)c1 N1(CCNC(=O)CC2CCCC(C(F)(F)F)O2)CCCNS1(=O)=O N1(C(COC(C)=O)=O)CC2(CC2)CC1C(=O)Nc1sc(C)nc1C C(=O)(CC1=CCCC1)NCC(CNC(=O)CC1CSCCS1)OC c1(C(=O)NC(CC=C)CNC(c2cnc(OC)s2)=O)ncnc(OC)c1F C1(CNC(C(C(C)C)SCC)=O)C2CCC(C2)N1C(=O)COc1cccc(F)c1 N(C(=NCCCC(C)(F)F)N(C)CCc1ncc(C)s1)C(CC)C CCCCCCC(CC)C(=O)N1CCCCC(CNC(=O)CC2CC3(CC3)C2)C1 CN1C(=O)CCCC1C(=O)NCC(C)(C)CNC(C12CC1COC2(C)C)=O C1(C(=O)NC(CCCC)C)CC2(CC(NC(=O)C(N)=O)C2)C1 NC1(CNC(N2CCN(c3ncccc3C(F)(F)F)CC2)=O)CCCOC1 Cc1nn(CC(=O)NCC(C)N(C(=O)C=CC(=O)NC2CC2)C)c(C)c1[N+](=O)[O-] C1(O)(CNC(C2(OC)CC2)=O)CCN(C(=O)CCc2cccnc2Br)C1 C(C)(C)(CCC(=O)N1CCOCC(NC(C2CC2(F)F)=O)C1)N(C)C CCCC(C(=O)N1CC2CC2C1C(=O)NCC12CC(CN1C)C2)C(C)C N1(C(C2C(C(=O)OC)CC2)=O)CC(C(=O)N(C2(CO)CC2)C)C(C2CC2)C1 c1(NCC2C(C)CN(C(=O)C3=CCCOC3)C2)ncc([N+](=O)[O-])n1C C(C(C)C(F)(F)F)N.Cc1nscc1C(=O)N(CCC(=O)N1CCCC1)CCO C12COCC1C(=O)N2.c1(CCCNC(C(C)=C2CCCC2)=O)cc(C)[nH]n1 C1(O)(CC(=O)NC2(CO)CN(C(C3CCC3c3ccccc3)=O)C2)CCCOC1 C1(C(=O)NCC(CC(=O)NCCOCCOCC)C)CC(=O)NC(=O)C1 CC(C)(C)C(C#N)C(=O)N1C(CNC(=O)COC2CCCOC2)CC2COCC12 N1(C(COCCCCC)=O)CCC2(CC2C(=O)NCc2nn(C)c(=O)o2)C1 c1(C(=O)NC2CCC(CNC(C3(OCC)CCC3)=O)C2)cnc(CSC)nc1O n1(CCC)cccc1C(=O)NC1CCC(CCNC(=O)Cc2n[nH]c(C)n2)C1 c1(C(=O)NC(C2CCCN2C(=O)CCC2(C)CC2)C)cc(-c2cnn(C)c2)no1 c1(C(N(C(CNC(CCSC)=O)C)C)=O)ccc2c(c1)N(C)CC2 N1(C(=O)OC(C)(C)C)CC(F)(CC#N)C1.C12OCCC1NC(=O)NC2.C(C)(C)(C)O C=CCCCC(=O)N1CCCC1C(C)(C)C(=O)NC(C)Cc1cccnc1 C1(OC)CCN(C(=O)C(C)N(C(=O)CCCNC(=O)OC)C)CC1 C(=O)(CC(C)(O)c1ccccc1)NCC1C(NC(C2(CCC)CCC2)=O)C1 NC1CC(F)(C(=O)NCc2c[nH]nc2C(=O)NCc2cccnc2)C1 c1(NCC2(C(N)=O)CCCCC2)cc(NC)nc(C)n1.C1C(O)CN1C.CS CC(=O)CCCC(C)C(=O)N1CC(C2CN(C(C3CCCSC3)=O)CCO2)C1 c1(CC)cc(NC2(c3nnnn3CCC3CC3)CSC(C)C2)cc(F)c1 C(C)(C(C(=O)N1CCOC(C)(CC)C1)C(C)C)NC(c1c(C)nc(CC)o1)=O CC1CCCCN1CCC(=O)NCCC1CC(NC(=O)C(C)N2CCCC2)C1 N1(C(CCCCC=C)=O)CC(C)CN(C(=O)CN(C)C(=O)OC)C(C)C1 C#CC(CNC(=O)CNC(=O)CCC1CC1C)CC(C)(C)C.c12ncoc1C2 Cc1ccc(OCCC(=O)NC2CC(=O)N(CS(C)(=O)=O)C2)c(Cl)c1 CCC(C(=O)N1CCC(C)(CNC(=O)CCCN2CCCCC2)C1)C(C)C CCC(CC)CCC(=O)N1CCCOC(CNC(C2CCCCS2)=O)C1 C1(NC(CC2C(CC)C2)=O)CC2(C1)CC(NC(=O)C(C)(C)Cc1cnn[nH]1)C2 CN1C(=O)CCC1CC(=O)NCc1cn(CC(=O)NCc2nccc(O)n2)nn1 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NCC(N1CCCCCC1)C Cc1nsc(C(=O)NC(C(=O)NCc2ccc(O)cc2)c2cccs2)c1N Cc1nc(C)c(CC(N2CC(CNC(=O)CCc3cccc(O)c3)CC2C)=O)s1 C1(CC(=O)NCCC2CCCC3CC23)CN(C(c2cncnc2)=O)CCO1 c1(C(N2C3C(NC(c4ccc(C(N)=O)o4)=O)CC(C3)C2)=O)ccc(S(N)(=O)=O)[nH]1 N1(C(CC)C)CC2CCC1C(N(C(=O)CCn1c(C)ccc1C)CC(=O)OC)C2 c1(OC)ccc(OC)c2sc(NC(=O)N(C)Cc3cccc4cnccc34)nc12 Cc1ccccc1-c1nc(-c2cncs2)nn1-c1nc[nH]n1 C(=O)(C(C)(C)C(C)(F)F)NC1CCN(C(c2ccc(-c3ccc(C)o3)s2)=O)C1 c1(C(N(C2CCN(C(C3C4(CC(OCC)C4)C3)=O)C2)CC)=O)nnc(O)nc1O N1(C(C2CC3(CC(C)C3)C2)=O)CC2CCC(C(=O)NCc3cnsc3)(C2)C1 N1(C(CCc2cc(C)ncc2)=O)CCC2(CCC(C(N3CCC3)=O)CC2)CC1 c1(OC)ccc(C(N2C(C(=O)NCC(c3ccccc3)O)CC3CC23)=O)c(Cl)c1 C1(N(C(=O)Cc2cn(C)nn2)CC)CCCN(C(C2CCCCCC2)=O)C1 C(=O)(C(O)C(C)(C)C)NCC(CNC(CSCC#C)=O)C c1(OC)cc(CC(=O)NCCCCC(C)NC(c2cncs2)=O)ccc1F N1(C(c2occ(C)c2)=O)CC2CCC1C1CN(C(=O)Cc3cncnc3)CC21 N1(C(CCC)=O)CCC2(C1)CN(C(C1CC3CCC1CC3)=O)CC(C)O2 CC(C)CCC(O)C(=O)N1CC(C(=O)NCC(C)(C)C2(O)CCC2)CC(C)C1 Nc1c(C(N2CCCC2C2(N(C(=O)C(O)CN(C)C)C3CC3)CC2)=O)ccnc1Br C1(N(C(=O)C(=O)NCC2CCCN2C(=O)NC)CC)CCCCCC1 C(C(Br)C(=O)NCC(F)CNC(=O)CC1(CO)CC1)NC(=O)OC(C)(C)C C1(CNC(c2c(C)noc2C)=O)CCC(C)CN1C(=O)CCC(F)F c1(C(N(C2CCCN(C(=O)CC3OCCO3)C2)CC)=O)ccc(C)c2ccccc12 C1(NC(c2ccc(OC(C)C)cc2Br)=O)CC(O)C12CCOCC2 N12CCC(F)(F)C(C1)C(=O)NC1(COC1)C2=O.c1(COC)cn2cccnc2n1 Cc1ncc(Br)c(N2CCC(O)C(C(=O)NC(c3ccccc3Cl)C)C2)n1 Cc1csc(C(=O)NCC2(F)CC(CNC(=O)C(C)O)C2)c1Br N1(C(c2ccc(SC)s2)=O)CC2(CCC2)C1C(=O)O C=CC1(C(=O)NC2CCCC(C(N)=O)C2)CCN(C(c2csc(C(C)=O)n2)=O)C1 Cc1c(-c2nn[nH]n2)cnc2c1N(C(=O)COCC1CCOC1)CCO2 N(C(=NCCc1ccccn1)NCCN1CC(C)OC(C)C1)CC(C(=O)OC)F Cn1ncc(C(N2CCN(C(=O)CN3CCCC3=O)CC2)=O)c1OCCC#N CC1C(NC(=O)CN2CCCCC2)C(C)CCN1C(C12CC=CC(C1)OC2)=O C1(NC(C(=O)N(CCCCC)C)=O)CCC(C#N)CC1 CN1CCCCC1CNC(C1C2CN(C(=O)C(O)C3CCCC3)CC12)=O C1(CNC(C(SC)SC)=O)(CO)CCN(C(=O)CSc2ccccc2C)CC1 C1(CNC(C2CCCC2)=O)CC12CCN(C(c1cc3c(s1)CCC3)=O)CC2 c1(C(N(CC(C)(C)NC(C(c2cccs2)SC)=O)C)=O)c(F)ccc(F)c1F C(=O)(C1CCCc2c(N)cccc21)N1C(C)(C)CC(NC(C2(F)CCCC2)=O)C1 N1(C(CCC=C)=O)CCC(C(N2CCSCC2C)=O)CC1CC N1(C(C(C)=CC2CC2)=O)CC(C)(C)OCC1CNC(c1cncc(F)c1C)=O c1(CC(=O)NC2CC(NC(C3ON=C(C)C3C)=O)CC2O)ccc(C)cc1C N1(CC(=O)NC2CCN(Cc3ccns3)CC2CO)C(=O)c2ccccc2C1=O C12(NC(C(C)C3CC3)=O)CCCCC1CN(C(=O)Cc1cncc(Br)c1)C2 C1(CCC)CN(C(C2CCC(O)C2)=O)CCN1C(=O)CC1CC1 C12(C(=O)NCCCC)CC(C1)N(C(=O)C(C)(C)CNC(=O)C=CC(C)C)C2 C1(C(=O)NCc2c(COC)nccn2)CNC(=O)CN1C(=O)CCC1OCCO1 N(C(=NCc1sccc1C)NC1CCCCC1)C1CCN(C(CC)=O)C1 C1(c2cn(CC(=O)NC(CC(=O)OC)C)nn2)CC2(CCCCO2)C1 Cc1nsc(C(N2CCCC2C=CC(=O)NC2CCCC2CCO)=O)c1N c1(C(N2CCC(C)(NC(c3ccc(OC)nc3)=O)CC2)=O)cc(Cl)c(F)cc1O C1(NC(CCOCCCOC)=O)CCC(O)CN(C(c2cnn[nH]2)=O)C1 c1(CC)ncc(C(=O)N(C)CC2CC(F)CN2C(c2cccs2)=O)c(C)n1 CC1(C)CCCOC1C(N1CCC(F)(C(=O)NCCOC(F)F)C1)=O C(C1=NOC2CN(C(C3CC=CC3)=O)CC12)NC(C1CN2CCCN1CC2)=O C(=O)(CC(C)C(F)(F)F)NCCC(C)NC(C12C(C(=O)OC)(CCC1)C2)=O c1(C(N2CC(C(C)(C)O)(CNC(=O)CN(C)C)C2)=O)cc(F)ccc1Cl c1(C(=O)NCC(C2CCOC2)NC(Cc2c(C)non2)=O)cc(S(N)(=O)=O)c(C)s1 CC1(C(N2CCOC(CCNC(C3CC4(CC4)C3)=O)C2)=O)CCC(O)CC1 C1(C2CCCN(C(=O)C=CCF)C2)(NC(C(C)(C)C(N)=O)=O)CC1 c1(C(N2CCC3CN(C(C4CN5CCN4CC5)=O)C3C2)=O)ccn2ccccc12 N1(C(COC(C)C)=O)CCC=C(C(=O)NC(C)CCN2CCCC2)C1 C(C)(N=c1[nH]c2cc(Cl)c(Cl)cc2s1)C1N(C(CCCCCC#C)=O)CCCC1 C1(NC(C(C)=C(CC)C)=O)CN(C(=O)CCn2cccc2)CC2(CCOCC2)C1 C1(F)(C(=O)NC2C(C(=O)NCCC3(COC)CC3)COC2)CC=CCC1 c1(OC)ccc2c(c1)C(C(=O)N1CCSCC(F)(F)C1)CCN2 N1(C(C(C2CCCCC2)N(C)C)=O)CCCC(NC(=O)COCCSC)CC1.C(CO)O N1(C(c2c(NCC)cccn2)=O)CCC(NC(=O)Cc2cncnc2)C(O)C1 C(O)(C(F)(F)F)C1(C(=O)NC2CCC2N2CCCC2)CCC1 N1(C(C2C(=C)C2)=O)C2CCC1C(NC(c1cccc(-n3nc(C)cc3C)c1)=O)C2 c1(C(=O)NC2CN(C(CCNC(N)=O)=O)CC(F)C2)nc2ncccn2n1 c1(NCC(C2CCC(=O)N2)(C)C)ccc2[nH]c3c(c2c1)CCCC3 CC1(CNC(C2CCSC2)=O)COCCN(C(=O)CCc2ncc[nH]2)C1 C(=O)(C(C)C(=O)OC)N1CC(C(C(=O)N(CC(O)COC)CC)O)C1 N1(C(C)C)CC(NC(C2(CNC(C3(n4nccn4)CC3)=O)CCCO2)=O)C(C)C1 C1(C(=O)NCC2COCCN(C(C(C)=CC)=O)C2)CCc2cnc(C)n2C1 C(=O)(C(C)CC(C)(C)C)N1CCC(C)C(NC(CN(c2ccccc2Cl)C)=O)C1 C#CCC(C(=O)NC(c1nc(C)oc1C)C)NC(c1csc(CC)n1)=O Cc1cc(C(N2CC3CC2C3NC(=O)CCc2ccc(Cl)s2)=O)cnn1 N1(C(C2CCC(=C)CC2)=O)CC2CCCC2C1C(=O)NC1CCOCC1C Cc1cc(N)c(C(=O)NCC(C)(C)CNC(=O)CCCn2ccnc2C)c(F)c1 C(=O)(C1=CCCSC1)N(CC(C)N(C(=O)CC1CC=CC1)C)C Cc1ccnnc1C(N1CCC(C)C1c1cn(C2CCCC2)nn1)=O c1(OC)ccc(C(=O)NCCC2(NC(c3ncncc3F)=O)CCC2)c(O)c1 c1(C(N2C(CNC(Cc3ncc(C)s3)=O)CC(C)(C)C2)=O)scc2c1OCCO2 N1(C(=O)CCn2cccn2)CCCC1C(C)(C)NC(C1CCC1)=O N1(C(C)=O)CCN(C(c2cc(C#N)c[nH]2)=O)CC1.C1(N)CCN(C(C2CSC2)=O)CC1 C(=O)(C1c2ccccc2C2CC1C2)NCC1(F)CCC(CNC(COCC)=O)C1 c1(C(=O)NC(=O)NCC(C)NC(CN(CC(C)C)C)=O)ccn(C(C)(C)C)c1 c1(C(=O)OCc2nc(C(=O)OC)c(C)o2)ccc(C(C)C)nc1F C1(CNC(C2CC(OC)C2)=O)CC2(CCN(C(C3CCC(F)C3)=O)CC2)C1 c1(CC(C)C)ccc(C(=O)OCc2nc(-c3ccc(F)nc3)no2)cc1 C(c1ccc(Br)c(Cl)c1)=CC(=O)NC(CNC(CCC)=O)CCOC C1(CNC(C2CSC2)=O)CC2(CCC2)CN1C(=O)CN1CCOCC1=O CN1CCC(C(=O)NCCC2CCC(NC(c3cc(Br)sn3)=O)C2)C1 C(C(C)NC(C1(CCF)CCOCC1)=O)(C(C)C)NC(c1cc(C)oc1)=O c1(C(N2CC3N(C(CC(C)(C)O)=O)C(CC3)CC2)=O)ccc(N)c2cnccc12 N1(C(C(C2CCOCC2)OC)=O)CC2CC2(NC(c2cc(F)n(C)n2)=O)C1 C1(C(N2CCCC(CNC(Cc3c(SC)cccc3)=O)C2)=O)CC(F)(F)C1(C)C c1(CC)cnc(C(c2nnnn2C(C)(C)C)NC2CC(C(F)F)C2)[nH]1 CCCC(CC)CCC(=O)N(CCNC(c1ccc2c(c1)C(C)CN2)=O)CC c1(OC(C2C(C)CCCN2C(=O)OC(C)(C)C)=O)ccc2nccnc2n1 c1(CN2C(C(=O)NC(C(C)(C)C)CO)CC(O)C2)ccc(Cl)cc1F O=C1CSc2ccc(C(=O)NC3CCC(NC(C4(O)CCSC4)=O)CC3)cc2N1 N1(C(=O)CC2CC3(CCC3)C2)CCCN(C(c2c(O)cccc2Cl)=O)CC1 N1(C(c2c(F)ccc(C)c2)=O)CCS(=O)(=O)C(CCNC(C2CC2C(F)F)=O)C1 C1(CNC(c2nn(C)c(C3CC3)c2)=O)CCCN(C(c2ccc(Cl)nn2)=O)CC1 c1(-c2scc(C(=O)NCCCNC(C3C(F)(C(=O)OC)C3)=O)n2)ccccc1Cl Cc1nc(C2CC2)[nH]c1C(=O)N(CC(C)NC(=O)C(C)SC(F)(F)F)C Cc1cc(=O)oc(C)c1C(NCP(C)(C)=O)(C1CCOC1)C.c12nnnn1CC2 c1(OC)ccc(C)cc1C(=O)NC(C)CCCNC(=O)C(CCO)N(C)C N1(C(C2N(CCC)CCC2)=O)CC2CCN(C(C3(C)CSC3)=O)CC12 C1(NC(C(C)OC2COC2)=O)CCC2CCN(C(c3cc(C(F)F)n[nH]3)=O)C1C2 Cc1nn(C)c(C)c1CC(=O)NC1CC(F)(CNC(C2CC=CC2)=O)C1 N1(C(C(CCC)C)=O)CCN(C(=O)C(C)(C)N(C)C)CC1CS(C)(=O)=O Cc1noc2ncc(C(=O)NC3CCC4CC3CN4c3cc(Cl)ncn3)cc12 c1(C(=O)NCC(CC)NC(c2cscc2F)=O)ccnc(Cl)c1OC c1(CC(=O)NCC(O)CCNC(=O)Cc2ccccn2)sccc1-n1cnnn1 C#Cc1ccnc(C(=O)NCC2(F)CCC(CNC(=O)C(C)CCOC)CC2)c1 C1(C(=O)NC(c2onc(CC(=O)OC)n2)(C)C)COC2(CCN(OC)CC2)C1 C1(CNC(C2(C)CC(NC(C3CC(OC)C3)=O)C2)=O)CCC(=O)NC1 Cc1nc(C(=O)NC2(CF)CCN(C(c3cccc(O)n3)=O)C2)ccc1Br c1(C(N(C(CNC(c2cc(C)cc(Cl)c2N)=O)C)C)=O)ccc2nnc(S)n2c1 c1(C(=O)NCC2N(C(C(CO)N(C)C)=O)CCCC2)ccccc1S(C)=O Cc1ccc(-n2ccc(C(N3CCSCC3C(=O)NCC(C)(C)O)=O)n2)cc1 C1(NC(c2scc(CNC(CNC3CC(C#N)C3)=O)c2)=O)CCC(F)(F)C1 C1(CN(C(c2ccccc2C2CC2)=O)CC)CCCCN1C(=O)CC1(CO)CC1 c1(NC(c2cc(Br)ccc2O)=O)n[nH]c2c1CN(Cc1ccc(Cl)o1)C2 N1(C(C(=O)NC(CC)(C)CCOC)=O)CCC(SC(F)F)C1 C1(NC(CC(CC)CC)=O)CC12CCN(C(c1ncnn1CC)=O)CC2 c1(C(=O)N(C2CC(N3CCC3)C2)C2CC2)nc(C2CC2)n[nH]1 N1(C(C(C2CCCCC2)C)=O)CCC(C)(C)C(C(=O)NCc2nncn2C)C1 c1(CC(=O)N(CC(C)NC(=O)Cc2csc(Cl)c2)C)cncn1C C12(C(=O)NCCNC(c3c(SC)cccc3)=O)C3C4C1C1C2C3C41C(N)=O N1(C(C(C)OC)=O)CCCC2(CCCN(c3ncc4c(n3)CCC4)C2)C1 Cc1c(C(=O)NC2CCC(C)N(C(=O)COC3CCC3)C2)cccc1Cl C1(CNC(C2CC(C)OCC2)=O)CN(C(=O)Cc2cccc(C#N)c2)CCN1C C12(CNC(C3ON=C(CC)C3)=O)CCC(C1)N(C(=O)Cc1c(F)cccc1Cl)C2 C1(NC(c2cnc(C(C)O)s2)=O)CC2(C1)CN(C(=O)CC(C)C(F)F)C2 C1(CNC(Cc2cn(CC)nc2)=O)CCCCN(C(=O)Cc2cccnc2)C1 Cc1c(C(N2CCC(C3CCN3C(=O)C=Cc3cnn(C)c3C)C2)=O)nn(C)c1N c1(-c2ccc(OCC)nc2)c(C(=O)NCc2ncon2)nn2c1CCCC2 C1(CC(=O)NCCC(COC)C)CN(C(=O)CN2CCCCC2C)CC1C c1(CN2CCCC(F)(CNC(C(C)C3CCC3)=O)C2)cccc2c1OC(C)(C)C2 N1(C(c2c[nH]c(=N)s2)=O)CCC(C(=O)N(C)C)(NC(C2CC(n3ccnn3)C2)=O)C1 C123CCC(C1)OC21CN(C1)C3=O.S(=O)(=O)(c1ccccc1)N1CC(NC(C)=O)C1 Cc1c(C(=O)NCCc2nc(C(N3CCC3CC(C)C)=O)co2)cncc1F C1(C)(CCC(=O)N(CC(O)CNC(C2CCCC2)=O)C)CC1(F)F N1(C(C2C(CC)CCC2)=O)CCC=C(C(=O)N(C2CCN(C)C2)C)C1 Cc1cc(C)c(C(N2CC(C(N3CC(C)(C)C3)=O)C(O)C2)=O)c(C)c1 CN1CCOCC1CC(=O)NCC(C1CCCO1)O c1(C(CNC(CSCC=C)=O)NC(=O)CSC2CCOC2=O)ccc(F)cc1F C12(C(=O)NC3CCCC(NC(c4c(NC)cccc4)=O)C3)CCC(C1)C(C)(C)O2 N1(C(C(C)(CO)N(C)C)=O)CCC(n2cc(CNc3ccccc3)nn2)C(O)C1 Cc1ccc(C=CC(=O)NCCCC(C)NC(=O)C(C)(C)c2cccnc2)s1 C(=O)(C(C(C)NC(=O)CCOCC(C)(C)C)C(C)C)Nc1cccc(OCC)c1 Cc1cc(=NC(=O)NCc2cn(C3CCCCNC3)nn2)[nH]n1CC(N)=O C1(N(C)C)CCN(N2CCC3(CCCCCC3)C2)CC1 C=C(C)C(C)(C)C(=O)NC1CCC1NC(C1(c2ccccc2)CC1)=O CC1(C(=O)Nc2ccc(-c3ccco3)nc2)CCN(C(c2ncccc2Br)=O)C1 N1(C(C(CCC)C#N)=O)CC(C)(C)C(NC(=O)C(C)n2cccn2)C(C)(C)C1 c1(C(N2CCC(CNC(C3CCC3C(F)(F)F)=O)C2)=O)ccc(C2CCC2)cc1 C1(CNC(COCCCC)=O)CN(C(=O)CCc2ccc(N)cn2)CCC1C CC(C)(O)CC(=O)NC1CC(O)(CNC(c2cn(CCCF)nn2)=O)C1 N1(C(Cc2c(C)ncs2)=O)CCC2CCCC12CNC(=O)CCCS(N)(=O)=O N1(C(C(CC)(C)C)=O)CC2(CCCN2C(c2cccc(OC(F)(F)F)c2O)=O)C1 C1(C(=O)NCC(C2CC2)OC)(NC(C2CC(SC)C2)=O)CCSC1 c1(C(=O)NC(CNC(C(CC)NC(N)=O)=O)CO)cc2cc([N+](=O)[O-])ccc2o1 c1(C(=O)NC2CN(C(c3n(CC)ncc3Cl)=O)CC(O)C2)cccc2ccnn12 c1(C(=O)NCCCCC(CO)NC(C2CC(OC)C2)=O)ccc2c(c1)CCCS2 C1(=CC(=O)NCC2(NC(C3C(C)=CCS3)=O)CC2)CCC(C)CC1 C1(NC(c2c(C)noc2)=O)CCC(CNC(c2cncn2C)=O)CC1 c1(CC)nc(CN(C(c2sccc2Br)C(=O)NC2COC2)C)cs1 C(=O)(N=c1cc(C)[nH][nH]1)C1N(C(c2ccc(C(=O)OC)cc2)=O)CC(F)C1 C#Cc1ccnc(C(=O)NC(C)(CC)CCNC(=O)C(CC)SC)c1 C12(CNC(CN(C)C3CC3)=O)CCCC(CN(C(=O)C(O)CSC(F)(F)F)C1)C2 C1(NC(CCc2cccc(-n3cc(CCN(C)C)nn3)c2)=O)CC2OCCCC12 C1(C(=O)NCC2(F)CC(NC(c3cc(C)c(Cl)s3)=O)C2)CCCC2(CC2)C1 C12(CNC(c3c(C)nn[nH]3)=O)CCC(CN(C(c3cc(=O)n(C)cn3)=O)C1)C2 C1(C(C(=O)NCC2C(C)CC3CC3C2)=O)CCC2CNCCC2C1 c1(C(N(CCCNC(C2C(CCC)CCC2)=O)CC)=O)cc(C)c(Cl)cc1F S(=O)(=O)(c1ccc(O)cc1)N1CCC(C(=O)NC2COCC2F)C(O)C1 Cn1cc(C(F)(F)F)c(Cc2ncccn2)n1.c12cccc(c1)CNC(=O)NC2 N1(C(CC2(CC)CCC2)=O)CC(NC(c2cnn(C(C)C)c2C)=O)CC2(CC2)C1 C1(C(N(CCn2cc(Cn3cccn3)nn2)CC)=O)CC2(CCC2O)C1 C#Cc1ccc(C(N2CCCC(C(=O)NCc3ccc(Cl)cn3)C2)=O)c(Cl)c1 N=c1[nH]cc(CNC(=O)C(=O)NCC2COCCO2)[nH]1 N1(C(CC(COC)C)=O)CCCC(NC(c2ccc(-n3ccnn3)cc2)=O)C1C C1(O)(CNC(=O)C(O)c2ccco2)CCCN(C(=O)C(c2ccccc2)O)CC1 C12(C(=O)NCCCCC(C)NC(c3ccccc3CO)=O)CC(C)(C1)OC2(C)C C(=O)(C1=CC2(CCOCC2)C1)NCC1N(C(c2cc(C(N)=O)oc2)=O)CCCC1 c1(OC)ccc(C(N2CCC(C)(C(=O)NCCCCN(C)C)C2)=O)cc1 c1(C(=O)NC(C(C)NC(C2(CC=C)CCCC2)=O)C)cc(C)ccc1[N+](=O)[O-] C1(CC)(NC(=O)CC#N)CN(C(=O)C(F)CC2CCOC2)C1 c1(-c2cc(OC)cc(C)c2)ccc2c(NC(C3CCS(=O)(=O)C3)=O)nsc2c1 C1(C)(C(=O)OC)CC(Nc2sc(Br)cc2F)CN1C(=O)C1CC1 c1(C(=O)NC(CNC(c2c(C)coc2)=O)C(C)C)c(Cl)ccc2c1OCO2 C1(C(=O)NC2CCC2CO)CN(c2ncncc2F)CCO1 Nc1c(C(N2CCC(F)(CNC(=O)C(F)=CC3CC3)C2)=O)cnc2ccnn12 c1(NC2CN(Cc3cccc(C)c3Br)CC2O)[nH]cnc2nc(Br)cc1-2 C1(OCC#C)CCN(C(c2c[nH]nc2CCNC(=O)C(COC)OC)=O)C1 Cc1ccnc2c(C(N3CCC4(NC(N5CCCC5)=O)CC4C3)=O)cccc12 C1(NC(C2(COC)CCCO2)=O)CC2CC(C1)N(C(=O)Cc1ccccc1F)C2 C1(O)(C(C(=O)NCC2CC3(CC3)C2)NC(c2c(C)nn[nH]2)=O)CCCCC1 C1(NC(c2ccoc2Cl)=O)CCCC(C(N2CCCC(CO)C2)=O)C1 C1(NC(C2CC23CC3)=O)CCC12CN(C(=O)C=CCCc1ccccc1)C2 C=C1CCCN(Cc2cnc(Cl)[nH]2)C1 N1(C(c2n(OC)cnc2C)=O)CC(NC(C2CC(C)C2)=O)C(C2CC2)C1 CC(C)C(CCc1ccccc1)C(=O)NC(CNC(c1ccsc1C#N)=O)CO C1(NC(CCC(N)=O)=O)CCOC12CCN(C(C1CCNC(=O)C1)=O)CC2 c1(C(=O)NCC(C)N(C)C(c2cccnn2)=O)cccc2cncn12 c1(N(CC(N2CCC(CO)C2C)=O)CCC)ccc(C)c(F)c1 c1(C(=O)NC2(C)CC(NC(C3(C)CC(=C)C3)=O)C2)cccc2c1C(=O)NC2=O c1(NC(c2nc(C(F)(F)F)cc(C)n2)=O)cc(F)cc(F)c1F C1(COC)CC(c2nnnn2C)(Nc2cnn(CC(F)F)c2C)CCO1 N1(C(CC2(OCC)CCC2)=O)CC(NC(=O)Cn2cccnc2=O)CC12CCC2 c1(CC)[nH]nc(C(N2CCC(=CCNC(C3CC3C(F)F)=O)CC2)=O)c1[N+](=O)[O-] CS(C)(=O)=Nc1cnn(CC(=O)NC2CN(C(c3sccc3Cl)=O)C2)c1 N1(C(c2nc(CC)sc2)=O)CCC2CCC(C1)N2C(=O)C(c1cncc(F)c1)C S(=O)(=O)(c1cc(C)cnc1NCC(C)CC1CC1)NCC=CCCC CCC(COC)(CC)C(=O)N1CC(C(=O)N(C)Cc2ncc[nH]2)C(F)(F)C1 C(C)(C)(CC(=O)N1CCCC(Oc2ccccc2)C1)n1cc(C(CC)(C)O)nn1 N1(C(C(C=C)CC)=O)C(C(N2CCC2C2CCC2)=O)CC2CCCC12 c1(C(N2C(CNC(=O)Cc3ccc(F)cc3Cl)CC2)=O)cc2c(nc1O)CCC2 C1(NC(CC=C(C)C)=O)C2CN(C(=O)C(C)(C)n3cccn3)CC12 C1(C2CCOCC2)(CNC(CCC=C)=O)CCN(C(=O)C(C(C)(C)C)N(C)C)C1 N1(C(c2ccc(CC)[nH]2)=O)CC2CCC1CN2C(=O)C(C)OC C1(C(=O)NCCCN(CCC)C(c2cccc(C(N)=O)n2)=O)CC12CCOC2 C1(c2nnnn2C2CCOCC2)(NCCNC(=O)OC)CSCCSC1 N1(C(CN(CC=C)C(C)=O)=O)CCC(N(C)C)CC1 S(=O)(=O)(c1ccc2c(c1)CC(=O)N2)NC(c1ccc(C(=O)OC)cc1)C(C)C CCCC(O)CC(=O)N1CC=CC(NC(c2cccc(SC)c2Cl)=O)C1 N1(N2CCC(=C)CC2C=O)CC(C=O)CC(C)(C)C1.C(C(Cl)=CCl)OC C(=O)(C1=NOC2(CCC2)C1)N1C(CC(=O)N(CCSC)CC)CC(O)C1 CCCCCC(F)C(=O)N1CCC(C(=O)NCCc2ccc(C)s2)(CO)C1 C(c1ccc(Cl)cc1F)=CC(=O)NCC12CC(NC(C(CCCC)O)=O)(C1)C2 c1(C(N2CC(NC(COC)=O)C3C2C3)=O)ccc2nnn(O)c2c1 CCCC(C(=O)N(CCC1CC1)CC1CC1)NC(=O)C(C)=NOCC#N CC(C)CC(C)C(=O)NCC1C(C)CCN1C(c1ccc(C2CC2)nc1)=O c1(NC(=O)NCC2N(C(C=CC=CCC)=O)CCC(C)C2)cc(F)c(C)cc1N C(=O)(CN=c1cc[nH]cc1)N1CC(C)OC(C(N2CCCC(C)C2)=O)C1 C1(NC(CC(C)(C)N)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)COCCO)C2 N1(C(C(CC)C#N)=O)CCC(C2CC2)(CNC(=O)CCOCC2CCC2)C1 N1(C(C=CCN(CC#C)C)=O)CC2(CC2)CC1CNC(=O)CCC1CC1C c1(NCc2c(C)non2)ncccc1S(=O)(=O)NC1CCC(C(N)=O)CC1 C(C(=O)NC1CC1NC(c1cncc(C(=O)OC(C)C)c1)=O)(C(C)C)OC(C)C N1(C(C2CCN(C)CC2)=O)CC(NC(=O)CSc2cnn(C)c2)CC(F)C1 C1(NC(C=CC=CC)=O)CCCN(C(=O)Cc2ccoc2)CC1 N1(C(C(CC#C)(C)NC(c2n[nH]c(C)c2Cl)=O)=O)C2CCC1CC1(CC1)C2 C1(CNC(=O)CC2C=CCC2)CCN(C(C2CCSCC2)=O)C12CC2 C(=O)(CCCC(=O)NCC1COCC1NC(c1cccc(C(F)F)c1)=O)N(C)C CCC(C)(O)C(=O)NC1CCCC1CNC(=O)CC1(N(C)C)CC1 C1(C(=O)NCC2CC2(F)Cl)CCN(C(C)(C)C)CC1.N12CC(C1)NC2=O C(C(S(=O)(=O)c1ccccc1)c1ccccc1)NC(C(C)C)C(=O)N1CCCC1 C(=O)(C(C)CC(C)(F)F)NCCCC1N(C(C(C)SCCCC)=O)CCC1 c1(OC)cccc(O)c1C(=O)NCCC1CCN(C(=O)CC2CC(F)C2)C(C)C1 c1(N2CCC(CC(N3CCCC(C(=O)OC)CC3)=O)C2)nc(Cl)nc2[nH]cnc12 Cc1cc(F)c(C(=O)NCC2CCCN2C(=O)COCCCF)c(Cl)c1 CC1CCN(C(c2ccn(C)c(=O)c2)=O)CC1C(=O)NOC1CCCC1 Cc1onc(C(=O)NC(C)C(C)NC(C2CCCCN2CC(F)F)=O)c1[N+](=O)[O-] C(=O)(CC(C)CC(C)(C)C)N(C(C)CNC(c1cnc(C2CC2)nc1O)=O)C C(=O)(CCCC(C)(C)CC)N1C(CNC(C(CC)OC)=O)(COC)CCC1 C1(CNC(c2c(CC)[nH]cc2)=O)CC2CCC1N(C(=O)CC(C)n1ccnc1)C2 CC1CN(C(C2(C)CCCO2)=O)CC2(CCN(C(=O)Cc3cccc(N)c3)C2)O1 C1(NC(C2(C)CC(F)(F)C2)=O)CC2CC(C1)N(C(=O)Cc1ccc(F)c(Cl)c1)C2 C12(C(N3CC(F)(CNC(c4n(CC)cc(Cl)c4)=O)C3)=O)CC(C)(C1)OC2(C)C C1(C(=O)OC)(C(=O)NC23CC(NC(C)=O)(C2)C3)CCCCC1.C1(=O)C(C)(C)N1 c1(CNC(c2cc(C(C)(C)C)n[nH]2)C)sc(C(=O)O)cc1Br c1(OC)cc(O)ccc1NC(c1c[nH]nc1CNC(c1nscc1C)=O)=O CC1CN(C(=O)CC2CCCNC2=O)CC(C)N1C(C1CC12CCOCC2)=O N1(C(c2c(C)nc(Br)s2)=O)CCN(C(=O)C(C)OCC(C)C)CC1CCO C1(=CC(=O)NCC2COCCN2C(C2COCCO2)=O)CN2CCC1CC2 C1(NC(CS(N)(=O)=O)=O)CN(C(=O)CC2CCCC2(F)F)C2(CCC2)C1 C(C1=CCN(CC(c2ccc(F)cc2)O)CC1)NC(c1c(C)snc1)=O c1(CNc2c(C(=O)Nc3ncc(C#N)cn3)nccc2)ccc2nc(O)[nH]c2c1 CCC(CC(F)F)C(=O)NCCOCCCNC(=O)Cc1cc[nH]c1 N1(C(=O)N(c2n[nH]c(C)c2Cl)C2CC2)CC2(CCCC2)C1c1ccccc1 O=C(C1CCCc2cncn21)NCC1C2CN(C(C3(CO)CCC3)=O)CC12 C12(C(N3CC(N(C(C(=Cc4cnc[nH]4)C)=O)C)C3)=O)CCC(CC1)C2(C)C C(CCC(O)C(=O)Nc1ccc(-c2ccc(C(F)(F)F)cc2)o1)N(C)C N1(C(=O)CC=Cc2ccc(F)cc2)CC(CNC(C2(F)CC2)=O)N2CCC1C2 CC1(C)CCC(CC(=O)NCC2(C)CCC(NC(c3ccnnc3O)=O)C2)CC1 C12(NC(c3cn(CC)nn3)=O)CCC(C1)N(C(c1[nH]nnc1C)=O)C2 CCCCC(F)(F)C(=O)NCC(CC(C)C)C(=O)N1CC(=O)NC(C)C1 C(=O)(CCC(=O)NC)NCCCOC.C1(C)(NC(C2C(=C)C2)=O)CN(O)C1 c1(CC(=O)NCCC(C)CCNC(c2cscn2)=O)cccc2ccoc12 Cc1cc2scc(CC(=O)NC3CCC(NC(C4CC4(F)C(=O)O)=O)C3)c2s1 c1(COC)cc(Cl)cc(S(=O)(=O)Cc2nc(C3CC3)nn2CC(F)(F)F)c1F c1(OC)cc(CNC2CCC(C(=O)NCC(C)(F)F)CC2)cc(F)c1F Cc1nc(O)ccc1C(=O)NC1C=CC(CC(N2C3CCCC2CC3)=O)C1 N1(C(C)=O)CCCCC12CCN(C(=O)NC1COC(C)C1)CC2 CCCCCCC(C)C(=O)NOCC(=O)NCCCc1nncn1C c1(OCC)ccc(-c2cc(C(=O)N(c3cnn(C)c3)CCO)ccn2)cn1 c1(C(=O)NC2CC(NC(c3c(C(C)C)ncs3)=O)C2)n[nH]c2c1CC(C)(C)C2 c1(CC)ccc(C(=O)NCC(CCOC)COC(=O)C2CC2)[nH]1 C1(OC)CCC2(C(=O)NC3(C(=O)NCCCN4CCCC4)CCC3)CC12 CC1CN(C)CCCN1C(=O)CCC1CCCN(C(=O)Cc2ccc(O)cn2)C1 CC(C)(F)C(C)(F)C(=O)N1CCC2C(C1)CN2C(=O)C=CBr c1(C(N2C(C(=O)NCc3ccc(C)c(C)c3)CC(F)C2)=O)c(O)ccc(F)c1F C(=O)(C(S(C)(=O)=O)C1CC1)N1CCC(NC(c2c(NCC)scn2)=O)CC1 c1(NC(N2CCN(CC(=O)NC3CCC(F)(F)C3)CC2)=O)cccc(Cl)c1 Cc1ccc(C(=O)OC(CC(F)F)c2ccccc2)cc1C(C)C C(=O)(C#CC(C)(C)O)NC1CCCC(N(C(=O)Cn2cc(C(F)F)cn2)C)C1 C1(CNC(C2C(C)C2)=O)CC2CCC(C1)N2C(C1(C)CC1(F)Cl)=O N1(C(C(CCC)OCC)=O)CC2CC(C1)N(C(c1cc(C#N)c(N)cc1O)=O)C2 c1(C(N(C(C)CNC(c2cn3cccnc3n2)=O)C)=O)cc2cc[nH]c(=O)c2s1 c1(C(=O)NCC(=C)CCNC(c2cc(N)cnc2Cl)=O)cc2c(C)cccc2[nH]1 N1(C(CC=CC)=O)CCOC(CN(C)C(C2CC3(CC3)CO2)=O)C1 c1(C(=O)OCC)nccnc1C(=O)N(C1(c2ccccc2)CCC1)CC N1(C(c2noc(CC)c2C)=O)CCCC(O)(CNC(=O)Cc2ccnc(O)c2)C1 C1(OC)CC(F)CN(C(c2cc(CNC(=O)C=CC(F)F)nn2C)=O)C1 C12(C(=O)NCC(C)(C)NC(C#CC(C)C)=O)CCCCC1NC(=O)C2 N1(C(C(=O)NCCOCCOC)=O)CCCN(C(C2C(C)(C)OC2(C)C)=O)CC1C N1(C(c2cncc(COC)c2)=O)CC2CCC1CC2NC(=O)C(C)S(N)(=O)=O N1(C(c2cnc(SC)nc2O)=O)CC2CCC(C1)N2c1nnco1 N1(C(C(c2ccc(F)cc2)OC)=O)CCN(C(c2ccccc2Cl)=O)CC(O)C1 c1(C(N2CC3CC(CNC(Cn4ccc(C)n4)=O)C3C2)=O)cc(F)cc(N)c1F c1(C(N2CCCC3(NC(CCC)=O)C(C2)C3)=O)cc(F)c(F)c(O)c1F CC1COCC(CC(=O)NCc2cc(C(=O)NC(CO)C3CC3)n(C)n2)O1 Cc1nccc(C(=O)NCC(O)CN(C(=O)C=CC2CC2)C)c1O C#CCC(O)C(=O)N1CC(C2CN(C(c3cnc(=N)[nH]c3)=O)CCO2)C1 C1(OCC)(CN2CCC2NC(=NCC)NCC(CC)CC)CCCCC1 CC1(C)CC(C(=O)NC2CCCC2(C)C)CN(C(C2CC(C)(O)C2)=O)C1 N1(C(C(C#C)(C)C)=O)CCCC(N(C(=O)C(C)CSc2ccc(Cl)cc2)C)CC1 CCCCCCC(C)C(=O)NCCC1(C(=O)N(CC(O)CO)C)CC1 c1(CC(CC(=O)OC)NCCC2CCSC2)ccc(F)c(Cl)c1 CC1=C(C(=O)N(CCCCCNC(c2cnn(C)c2C(C)C)=O)C)CC1 C1(NC(C2CCSC2)=O)CCCCN(C(c2ccc(-c3ccccc3)[nH]2)=O)C1 N1(C(C2C(CNC(c3occ4c3CCC4)=O)OCC2)=O)CCCC(F)CC1 C(=O)(C#CC(C)(C)C)NC1(C(=O)NCc2n(C)nnc2)CCSC1 c1(C(N2C(C)C(NC(C3(C)CCCC3C)=O)CCC2)=O)cc2c(nc1O)CCC2 C1(NC(c2ccc(-n3cc(Cl)cn3)c(Cl)c2)=O)CCc2nnc(O)n2C1 O=C(CCN=C(NCC1CC1)NC1CSCC1C)N(Cc1ccc(F)cc1)CC1CC1 Cc1cc(C(N2CCN(C)C(CNC(C3CCCCC3(F)F)=O)C2)=O)cc(N)c1 C(=O)(C(CC)C(=O)NC(c1cn(C(C)(C)C)nn1)C)OCC c1(C(N(C2CCCN(C(C3(OC)CCCCC3)=O)C2)CC)=O)cn(C)c(O)n1 C1(C(=O)NC2CCCN(Cc3cnc(Br)s3)C2)CCc2cc(Br)ccc2O1 C1(n2ncc(NC(C(=O)NCCOCCNC)=O)c2)CCS(=O)(=O)C1 C1(CC(=O)N(CCC(C)NC(=O)C(c2ccccc2F)F)C)CCOC1(C)C C1(CC=C)(C(=O)N(C)CC2CC2(C)C)CCN(C(=O)CCC=CC)C1 C(C)(C)(C(=O)NCc1cc(C(=O)NCC2=CCCC2)no1)OC C1(C(C2(CNC(=O)C3CC3)CC2)C)CN(C(=O)OCCc2ccccn2)CCO1 CC(C)CC(C(=O)NCC(C1CC1)N(C)C)ONC(=O)CCc1nccn1C C1(C)(C(N2CCC(O)(CNC(CC3(OCC)CC3)=O)C2)=O)CCN(C)C1=O C#Cc1ccccc1CC(=O)NC1(C(=O)NCCC2(C)N=N2)CC1C CC1=NS(=O)(=O)N(C)C=C1C(=O)N(CCCNC(c1cc2c(nn1)CCC2)=O)C Cc1ncc(C(=O)NCC2CN(C)CCN2C(c2nccs2)=O)c(C)n1 C(N=c1[nH]c(=NCCNS(=O)(=O)C(F)F)c2sccc2[nH]1)C1C(C)(C)OCCO1 C#Cc1cncc(C(N2CC(OCCNC(c3ccnc(S)c3)=O)C2)=O)c1 C1(NC(=O)CC2SC(=N)NC2=O)CC2(C1)CC(NC(=O)Cn1ccnc1CO)C2 c1(C(N(C2CCN(C(C(C)N(C(N)=O)CC)=O)C2)C)=O)ncccc1OC(F)F CC(C)(C)CCC(=O)NCC1CC1NC(c1ccc(-c2cccs2)cn1)=O Cc1ccc2c(c1)C(CN(C)CC1CC3C(C1)C3(C)C)CC2 c1(C(=O)NCCc2onc(CCCOC)n2)ccccc1-c1nc(C(C)=O)no1 O=C1CCC(CC(=O)NC2(CNC(=O)CC3CCO3)CCC2)N1 C=Cc1cnn(C)c1C(=O)NCC(C)N(C)C(c1coc(SC)c1)=O N(C(=NCCCNC(C)C)NCCC1CCCO1)Cc1c(CC)cccc1 c1(C(N2CCC(NC(CSCCOC)=O)C2)=O)ccc(Cl)cc1Br c1(OC)nccc(C(=O)NC2CCC2NC(=O)C(C)NC(N)=O)c1F C1(C(=O)Nc2ccc(F)cc2)CC12CCN(C(c1cccc(Cl)n1)=O)C2 C1(CNC(C(C)OCCOCC)=O)COCCN(C(c2cn(C)cc2C)=O)C1 C1(C(=O)Nc2scc(S(=O)(=O)NC)c2)Cc2cncn2C(=O)N1 CCC(C)(C)C(O)C(=O)N1CCCC(CN2CCN(C(=O)CC3(C)CC3)CC2)C1 N1(C(C(C)SCCCC)=O)CCCCC12CN(C(=O)Cn1cncc1C)C2 c1(CCC(=O)N(CCOC)CCNC(=O)Cc2cncn2C)ccc(Cl)c(F)c1 C1(CNC(C2(NC(CCCN(C(C)C)C)=O)CC2C)=O)CC2CC1CC2O c1(NC(C2(C#C)CN(C(=O)C(C)c3ccsc3)C2)=O)cc(C#N)ccc1O c1(C(N2C(C(=O)NC(CC)CCOC)CCC2)=O)cnc(S)nc1 CCC(F)C(=O)NCC(C)CN(C(=O)CCSCc1ccccc1)C C(=O)(CC(C)(C)C(=O)NC1CCCC1C(=O)NC1CC2(CCC2)C1)OCC c1(CNC(C(CCC)OCC)=O)nnc2n1CCN(C(C1CC1F)=O)C2 c1(CC)cccc(C(=O)NCC(C)=CC(=O)NC(c2cnc(C)s2)C)n1 c1(C(c2nnnn2C2CC(F)(F)C2)NCCCC=C)ccc(Cl)c(C)c1OC C(C1=NOC2(CCC2)C1)NC(CC(C1CC1)NC(=O)OC(C)(C)C)=O c1(C(=O)NC2(CC=C)CCN(C(c3cnc(C)cn3)=O)C2)cc(C)c(Cl)cn1 C1(C(=O)Nc2c(OC)nccn2)CC12CCN(CCc1ncc(Cl)cc1Cl)C2 C1(C)(C(=O)NCCCN(C(c2ccc(C3CCCC3)cc2)=O)CC)CC2CCC1C2 N1(C(C=C(C)C(C)C)=O)CCN(C(C2CC2C(C)(F)F)=O)C2(CC2)C1 CC1(C)CCC(C)(C(N2CCC(CNC(=O)C(c3cccnc3)O)C2)=O)CC1 c1(NC(=O)C=C2CCN(Cc3scc(Br)c3Br)CC2)cc(O)nc(O)n1 c1(N2CC(NC(c3cccc(C(C)=O)n3)=O)C(C)C2)nnc(C)c(C)n1 C1(CNC(c2scc(C)c2)=O)CN(C(c2cnc(C(C)C)s2)=O)CCCO1 N(C1CS(=O)(=O)Cc2ccccc21)Cc1c(C)c([N+](=O)[O-])cc(Br)c1 N1(C(C(C)OCCC=C)=O)CCC(NC(C2CC2F)=O)C(OC)C1 Cc1cc2ncn(CC(C)Oc3ccc(Cl)cc3Cl)c2cc1C CN1CCC(CC(=O)NC2CC23CC(NC(c2cnn(CC4CC4)c2)=O)C3)C1=O C1(O)(CNC(C(Cc2c(C)noc2C)C)=O)CCN(C(=O)C(F)=CCCF)CC1 CC(CN(C)C)CCC(=O)NC(C(=O)NOCCN1CCCC1=O)C1CCC1 N1(C(C(C(C)C)C)=O)CC2(CCCC(CNC(C3CC(N(C)C)C3)=O)O2)C1 C1(C(=O)NC2(C)CCSC2)CN(C(c2cccnc2O)=O)CCO1 N1(S(c2cccc(C(=O)OC)n2)(=O)=O)CC=C(c2cc(C)cc(C)c2)CC1 n1(CC)ncc(Cl)c1C(=O)NC1CCCC(CN(C)C(c2n[nH]c(C)c2F)=O)C1 N1(C(C(=O)N(C2CCC(C(=O)OC)CC2)C)=O)CC2CCC(OC)C2C1 N1(CCC)CCCC(C(=O)NCC(CCOC)NC(=O)COCC(C)C)C1 C(=O)(CN=c1cc(C)nc(N2CCC(C(=O)Nc3ccccc3)CC2)[nH]1)NCC C1(NC(c2n[nH]c(C)c2C)=O)CN(C(=O)C(O)CC(C)(C)C)C2CCCCC12 C=C1CC2CCCC(C1)N2C(=O)C(C1CCN(C(=O)C(CC)OC)CC1)C Cc1ncnc(C)c1OCC(=O)NC1CCC(C)N(C(C2CC(=C3CC3)C2)=O)C1 CC(C)CC(C(=O)N(CC(C)(C)N(C)C)C)NC(=O)C(=O)C(C)C C(CCCCC(=O)N1CCC(C(CC)CC)C1)N(C(CCSCCC)=O)C CC1CCN(C(=O)CCc2cccc(Br)c2Cl)CC1NC(C1(C)CC1)=O C(C(CC(C)C)C(=O)NCC(=O)N(C)C)NC(CC1N(C)CCCC1)=O O=C(C1Cc2c(Cl)cccc21)NC(C1CCOC1)CNC(=O)CC1CCC1 C1(NC(C2CCN(C(CC)=O)C2)=O)CC2(C1)CN(C(c1csc(Cl)c1)=O)C2 N1(C(C2C(C=C)C2)=O)CCC(CC(=O)NCCc2cc(C)no2)(C(=O)OC)CC1 CC1CC(NCc2cnc(Cl)n2C)C(=O)N1c1cnn(C)c1 c1(C(=O)NCC2C(NC(C3C(C(=O)OC)CC3)=O)C2)ccc(F)cc1Cl c1(C(C(N2CCC(CNC(C(C)(C3CC3)OC)=O)C2)=O)=O)cc(F)cc(Cl)c1 c1(C(N2CC3C(NC(C#C)=O)C3C2)=O)cccc(C(F)(F)F)c1CC Cc1cc(NC(C2CC2CNC2CCC(CO)CC2)=O)ccc1Cl C1(C#N)(C(=O)NC(C)CNC(c2nn(C)cc2CO)=O)CCc2ccccc2C1 c1(C(=O)NC2C(CNC(CN(CCOC)C)=O)CC2)sc(C)nc1C(F)(F)F C(=O)(CCCCCCCBr)N1C(CC)CN(C(=O)C(C)(CO)CO)CC1 C1(OC)(CNC(C2(OC)CC2)=O)CCCN(C(C2COCCN2CC(F)(F)F)=O)C1 c1(C(N(C2CCN(C(C)=O)C2)CCC)=O)ccc(C(=O)NCC2CC2)cc1 C(CCCCCC(=O)NCC(CC)(CC)C(N)=O)NC(CCSCCCC)=O C1(NC(COC)=O)CCC(C)(CNC(c2cnn(C)c2N)=O)CC1 N#Cc1c[nH]ccc1=NC(CNC(=O)NC1CC1c1ccccc1)CO C12(NC(C(=O)NCC(C)C(=O)O)=O)COCC1CN(C(c1cccs1)=O)C2 Cc1cc(C(=O)NCC2CCCC2NC(=O)Cc2cnn(C(C)C)c2)c(C)o1 C1(N(C23CC(C(=O)OC)(C2)C3)C(C#CC)=O)CC2CC1CN2 Cc1oc(C(F)(F)F)nc1C(=O)NC(C)(C)CCN(C(=O)CCC1CCOC1)C C(CC(C(=O)N1CC2CCC2C1)NC(=O)CC(C)(C)SC)SC CC(CCC(C)(C)C)C(=O)NCC(=O)NC(C1CC(=O)C1(C)C)=O Cc1noc(C)c1C(C)C(=O)N(C)CCNC(c1cc(Cl)nn1C)=O Cc1cc(C(N2CCC(NC(=O)CC34COC(C(F)(F)F)(C3)C4)C2)=O)nc(C)c1 Cc1ncnc(C)c1CC(=O)N(C)CCOCCCN(C)C(C1CCOCC1)=O N1(C(CN(CCC#C)C)=O)CCCC1(C(=O)NCCC(COC)OC)C(C)C C1(C(=O)NCCC2CC(C(=O)NC(C)CC3CCCC3)C2)(CO)CCOC1 c1(C(N2C(CNC(=O)OC)CC2)=O)ccc2c(c1)COCC2 C(S(=O)(=O)c1ccccc1)c1ccc(OCC)s1.C12CN(CC1NC(C)=O)C2=O N1(C(c2c(C(C)C)n(C)nc2)=O)CCCCCC(NC(=O)COc2ccsc2)C1 c1(C(=O)NCc2ncc(C(F)(F)F)[nH]2)cc(F)c(F)cc1Cl.C12=CCN(CC1)CC2 c1(C(=O)NCCOC(CNC(CC2(C)CCC2)=O)(C)C)cc(=O)n2nccc2[nH]1 Cn1cc(CC(C(=O)O)C(c2cnn(Cc3ccccn3)n2)=O)cn1 C(=O)(CCC(O)C(C)(C)C)NC(CNC(CCN1CCC(C)CC1)=O)C1CC1 c1(NC(C(=O)NCc2c(CC)cccc2)=O)cc(F)c(F)cc1F CC1CC(NC(=O)CCC2OCCO2)CN1C(C)C(=O)Nc1ccccc1 C1(C(=O)NC2CN(C(C(C)(C)F)=O)CC2O)C2CC(F)(F)CC12 C(CCC)(C(O)C(=O)NCC1([Si](C)(C)C)CC1)NC(CCCCCC)=O c1(C(=O)NCCC(C)NC(c2coc(Cl)c2)=O)cc2ccc(O)cc2n1C c1(C(=O)NC2CC(O)(CNC(C(C)NC(CC)=O)=O)C2)cc(OC)c(OC)c(N)c1 C1(C(C)NC(Cc2ccco2)CO)CCN(C(=O)C(C)C)CC1 C=CCC(C)C(=O)N1CCC(N(C(=O)CCCn2cccn2)CC2CC2)CC1 C1(NC(C23CC(C)(C2)C3)=O)CCN(C2CC2)C1=O.c12nc(cs1)CNC2=O CCC(C(=O)NC1CCC(NC(=O)C=C2CCC2)C1)NC(N)=O C1(C2C(C(=O)NCC34CC(c5ccccc5)(C3)C4)C2)CCCN1S(=O)(=O)CC C1(CC(C)C)CCC(NC(=O)CCN(C(=O)CN2CC(C)(C)C2)C(C)C)CC1 Cc1nc(C(N2CCCC23CCN(C(=O)CC2C=CCC2)C3)=O)c2ccccn12 C1(C(N(C(C2CN(C(C(=O)NCCC)C)C2)C)CC)=O)CCNC(=O)C1 N1(C(CC(CC)O)=O)CCC(O)C(C(=O)Nc2ccc(O)cc2C(N)=O)C1 N1(C(C(OC)OC)=O)CCC2(CCC(NC(c3ccc(F)c(Cl)c3)=O)C2)CC1 C=C(C)C1OCCC1C(=O)N(CCC(=O)Nc1cccc(C(C)C)c1)CC1CC1 c1(CN2CC3C(C(=O)Nc4cnc(OC)nc4)C3C2)cccc(S(C)(=O)=O)c1 c1(C(=O)NCCOCCCNC(C(C)n2cncn2)=O)ncnc(O)c1F c1(C(C)=O)ccc(O)c(S(=O)(=O)N(c2ccc3c(c2)CCC3)C)c1 Cc1cc(O)n2ncc(C(=O)NC3CC(CNC(C4CCN(C)CC4)=O)C3)c2n1 O=C(C(O)C1=CCCCC1)NC1CC(NC(c2ccn(CC(F)F)n2)=O)CC1O C1(CC)COC(CC)CN1C(=O)C(=O)NCc1cc(Cl)cnc1C CC1(C)CCN(CCNC(C2CC(n3cc(CC4COC4)nn3)C2)=O)C1 CCCCCC(C1CC1)NC(=O)CCN(C(C1(C)C=CCCC1)=O)C1CC1 Cc1c(Br)ccc2[nH]c(C(=O)Nc3ccnc(OC(C)C)c3)cc12 c1(C(N2CCC(C)(NC(=O)C(=O)NC3CC3)C2)=O)cc2cccn2c(O)n1.CN c1(OC)cc(F)c(-c2ccc(CNC(=O)CC(F)(F)F)cc2)cc1F c1(CC(N2CCC(N(C(=O)CCCCCF)C)C2)=O)ccc2ccncc2c1 C(=O)(C(C)(C)C(N)=O)N1CC(CC)SCC1.C(=O)CC(O)CN N1(C(c2c(OC)cnnc2)=O)CCOCC(C(=O)NC2CCCC(CO)C2)C1 C(=O)(C(C)(CC)CO)Nc1[nH]nc(-c2ccc(OCC)cc2)n1 c1(C(=O)NCc2occ(C)n2)nc2ccccn2c1-c1ccn2cnnc2c1 Cc1cnc(C(=O)NC2CCCN(C(c3cc4c(s3)CCCC4)=O)C2)cc1C#N C=C=CC(C)C(=O)NCC1CC1C(=O)NCc1cn(C)cn1 CC1CC(CNC(=O)C(C2CC=CCC2)NC(c2cnnn2C)=O)=NO1 C12(C(=O)NCC3N(C(C4N(CC)CCC4)=O)C4C(C3)C4)CC3CC(C(=O)N1)C2C3 N1(C(=O)NC)CCC(Oc2ccccc2NCCS(C)=O)CC1 N=c1ccc(CNCC23COC(NC(=O)COC4CC(F)(F)C4)(C2)C3)c[nH]1 C(CC(CC)C(=O)NCC1CC(F)(CNC(c2n[nH]cc2Cl)=O)C1)=CC C1(NC(CC(=C)C)=O)CCCCC12CCN(C(=O)Cc1ccc3c(c1)CCC3)C2 c1(C(N2CC(COC)N(C(=O)C=C(C)C)CC2)=O)ccc2cccc(O)c2c1 C1(CNC(c2cn(CC(C)C)nc2)=O)(CO)CCN(C(c2csc(=N)[nH]2)=O)C1 N1(C(CC=CCC)=O)CC2CCC2(C(=O)NCc2cc(C)co2)C1 N1(C(c2cncc(C)c2C)=O)CCC2CN(C(c3cccc4occc34)=O)CC12 C(=O)(CCN=C(NCC1CCC2(CCC2)CC1)NC(C)C1CC1)NC N1(C(C2(OC(C)C)CCC2)=O)CCN(C(C2CCC(=O)C2)=O)CC(O)C1 C1(C(=O)Nc2cnn(C(C)C)c2)(CC)CCCN(C(=O)C(C2CC2)OC)C1 N1(C(C2C3N(C(C(CCOC)OC)=O)C(CC3)C2)=O)CCCC(O)(C2CC2)C1 CC1C(C(=O)NC2COCC(C)(C)C2)CCCN1C(=O)Cn1cncn1 c1(CNC(C2(NC(C)=O)CC2(C)C)c2n(CCC)nnn2)cccc(OC)c1 C(C(COC)C(=O)NCC(N1CC(C)(OC2(C3CCCOO3)CC2)C1)=O)OC C(=O)(C1=CC2(CCN(C(=O)C(CO)C(C)(C)C)C2)C1)NCC(CN(C)C)(C)O C(C(C)C(=O)NC(C1(C(N2CC(O)(CCO)C2)=O)CC1)C)OC CCCCCC(O)CC(=O)NC(CNC(c1cc[n+]([O-])cc1)=O)CO c1(CC(=O)NC2C(NC(C(C3CCC3)OCC)=O)COC2)cccc2sccc12 Cc1coc(C=CC(=O)N(C)CC2(O)CN(C(C3CCCOC3)=O)C2)n1 CC1SCCCC1C(=O)NC(c1cnn(C)c1)C(=O)NCCOC(F)F C1(C(=O)NC(C)CC(=O)NCCc2nncs2)CCCC(C)(C)C1 Cc1ccc(C(C)NC(=O)CC2CN(C(=O)C3=NOCC3)CC2C)cc1 FC1(F)CCC(n2nc(Cc3ccccc3)nc2-c2ccc(Br)cc2)C1 C1(C(=O)NCC(CNC(=O)CCOCC(F)F)F)CC2(CCCC2)CO1 CC1(C)CCCN(C(c2cccnc2)=O)C1CNC(C1CC12CC2)=O N1(C(c2n(C)ccn2)=O)CCC(C(=O)Nc2nc(F)ccc2Br)C(O)C1 C1(CNC(C(=O)NC2C(SC)CCC2)=O)CCCCC1Oc1cccc(Cl)c1 N1(C(C2(NC(C(CC)C(C)C)=O)CSC2)=O)CCCCCCCC1 C1(CNC(=O)Nc2ccn(CC(=O)O)c2)CC2CCCN2C1 N1(C(CC(=C)C)=O)CC(NC(=O)CCCN(C)C(C)=O)C(C)C1 C=CC(CC(=O)NC(C)(CNC(c1c(C)coc1CC)=O)CO)c1ccccc1 c1(OC)cc(C)sc1C(N1CC(CCNC(=O)CCC(C)N(C)C)C(C)C1)=O c1(C(N2CCN(C(COC(C)=O)=O)C3C2C3)=O)cc2ccncc2c(O)n1 Cc1oc(C)c(C(N2CCC(C(N3CCC(OCCF)C3)=O)C2)=O)c1C n1(CCC(=O)NC2(C)CC(NC(CNC(CC)=O)=O)C2)nc2ccccn2c1=O CC#CCCCC(=O)NCC1CC1NC(C1CN(CCCSC)CCO1)=O CCC(CC(=O)NCCCCNC(c1cccc(CS(N)(=O)=O)c1)=O)SC c1(C(C)C)nc(NCC(N2CCCC2)C)cc(=NC2CC(=O)N(CC3CC3)C2C)[nH]1 C(C1=CCN(C(=O)C(N2CCC(C)C2)=O)CC1)NC(c1cnc(CC)nc1)=O C(=O)(C1=CNC2=NCCC2=C1)NC1CC(C(N(C)Cc2n(CC)cnn2)=O)C1 CC1CC(C(=O)NC(C)CNC(C2(c3ccno3)CCC2)=O)CC(C)C1 Cc1[nH]nc(C(=O)NCC2C3CC2N(C(C2CCC4CC4C2)=O)C3)c1Cl c1(NCC2OCCN(C(C(CCC)NC(N)=O)=O)C2)ncnc2onc(C)c12 C(=O)(C(O)CCC(F)(F)F)N1CC2(CC(NC(=O)Cn3cnnn3)C2)C1 C1(C(N(C(C)CS(C)=O)CC)=O)CC(C(C)(C)C)CNN1C(=O)OC(C)(C)C Cc1cccc(Br)c1C(=O)Nc1ccc(Cn2cc(CC(O)C(C)C)nn2)cc1 c1(C(=O)NCCC(=C)CNC(c2cnc(OC)nc2)=O)cnc2c(c1)CCC2 CC(=O)CCC(=O)N1CCCC1C=CC(=O)NC1CC(N2CCCC2)C1 C1(C(=O)NCCOCCNC(CCCC=C)=O)CS(=O)(=O)CC12CCC2 c1(C(c2nnnn2CCC2CC2)NC(CC)C(C)C)cccc(O)c1 c1(N(CC)CC)ccc(C(N2CC(CCCCNC(=O)CS(C)(=O)=O)C2)=O)cn1 Cc1c(C(N2CCC(NC(=O)C(C)n3cnnn3)C2(C)C)=O)cnc2nncn12 C1(NC(C(CC=C)C)=O)CC2CN(C(c3ncoc3-c3ccon3)=O)CC12 c1(OC)ccc2c(c1)C(C(=O)NCc1cscc1C)CCC2 CC(CCC(=O)NCc1ccc(CNC(C2(C#N)CCC2)=O)cc1)N(C)C C=CC1(C(=O)NCC2CCCC(NC(C3(CC)CCC3)=O)C2)CCCCC1 c1(CC)ccccc1C(C(=O)Nc1cccnc1)N(CC(C)C#N)C CCCC(CNC(c1ncncc1C)=O)C(=O)NC1CC(Cl)(Cl)C1 c1(C(=O)NC2C(NC(C(C)(C)F)=O)CCCC2)ccc(Br)cc1[N+](=O)[O-] C1(OC)CN(N2CCC(NC(=O)OC(C)(C)C)CC2)CC1c1cnn(C)c1 Cc1n[nH]c(C)c1C(c1nnnn1C1CCCC1)NCC1CC1CC1CCC1 N(C(=NCCSCC)NCC1(F)CC1)CC(=C)Cl c1(N(CCCC)CCOC)cc(S(=O)(=O)NCC2CCC2)ccc1C#N C=CC1(C(=O)NCCC2(O)CCOC2)CCN(C(=O)CCc2nccs2)C1 C1(CNC(C(C)n2cncn2)=O)C(C)CCN1C(C1COC(C)(C)C1)=O C(=O)(CCS(N)(=O)=O)NC(CCNC(c1nc(C(C)OC)sc1)=O)(C)C c1(CN2CCC(NC(c3cc4cccnn4n3)=O)CC2)c[nH]c2ccc(Br)cc12 Cc1cc(NC2CC(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2(C)C)n2nc(C)nc2n1 C1(NC(C2CCN(C)C2=O)=O)CCCC(NC(=O)CCN2CCC2)CC1 NC1C(c2ccccc2)CN(Cc2c(Br)ccc3ncccc23)C1 C(=O)(C1=COCCC1)N1CCC(O)(CNC(C(C(C)C)n2cnnn2)=O)C1 C1(NC(c2cc(OC)c(O)cc2)=O)CN(C(c2cc(C)n(C)n2)=O)CC(C)(C)C1 N1(C(C(C)(C)O)=O)CCC2(CC1)CC2NC(C1CCCN1N=O)=O N1(C(CCSC)=O)CCC(C)C(NC(c2c[nH]nc2Cl)=O)C1 CCCC(O)C(CO)NC(C1CC2CCC1N2C(=O)CCCC1CC1)=O c1(C(=O)NC2C(NC(Cc3cncc(C)c3)=O)CCC2)cncc(N)c1C c1(C(N2CCC(=CCNC(C3C(C(C)O)C3)=O)CC2)=O)c(Cl)cc(Cl)nc1N c1(C(N(CCCCNC(=O)C(O)C2CC2)C)=O)ccccc1Br C1(C(=O)OC)CCCC(n2cc(C3CCN3C(c3cnn(C)c3C)=O)nn2)C1 c1(C(=O)OCC)cccc(NNC(=O)N2CC3OC(=O)OC3C2)c1Cl C1(CO)CCN(C(C23CC(CCNC(C=Cc4scc(C)n4)=O)(C2)C3)=O)C12CCC2 c1(SCCC)nc(C)cc(NC(=O)NCCCCN2CCC2)n1 Cc1ccn(C(C)C(=O)N(C)CC2(O)CN(C(=O)COC3CC(F)(F)C3)C2)n1 C1(C(=O)NCC(CC)NC(c2c[nH]nc2C2CCCO2)=O)CCC(=O)N1 CC1CN(C(C2C3CCOCC23)C(=O)Nc2ccccc2Cl)CC(C)S1=O C(=O)(C#CC1CCCCC1)NCC(C(N1CCC(C(C)C#N)CC1)=O)(C)C N1(C(CN(C(=O)OCC)C)=O)CCCC2(CNC(c3oncc3C)=O)CC12 C1(C2CCCC2)(C(=O)NCC(C)NC(=O)C(O)CC2CC2)CCNC1=O N(C1CN(C(c2cnn(C(C)(C)C)c2)=O)Cc2ccccc21)C(CC(C)(F)F)=O C12(C(=O)NCCN(C(C(C)SC)=O)C)COC(C1)C2 N1(C(c2ccc(C)nc2)=O)CC2(CC(NC(=O)Cc3ccc(Cl)c(C)c3)CO2)C1 C1(NC(CCC=C)=O)CN(C(c2cc(C#N)ccc2Cl)=O)CC1S(C)(=O)=O C(=O)(C(Cn1cccn1)NC(C1CCSCC1)=O)N(C)Cc1ccccn1 C1(O)(CC(=O)N(CCC)CCNC(=O)C(F)=CCCF)COC(C)(C)C1 C1(CNC(c2c(C)nn(CC)c2C)=O)CN(C(=O)CC(C)O)CC2(CCC2)O1 c1(CC)cc(C(=O)NC(CO)C(C)NC(c2sccc2SC)=O)ncn1 N1(C(C2OCCC(C)C2)=O)CCN(C(c2ccc(=O)n(CCO)c2)=O)C2CCC12 N1(C(C(CC)=CCCC)=O)CC(C(=O)NCC2(CN=[N+]=[N-])CC2)CC12CCC2 C1(NC(C(C)OC)=O)C2CCC1CN(C(c1ccc3c(c1)OCO3)=O)C2 c1(CCC)c(C(=O)N(CCCOCCNC(=O)CCn2ccnn2)C)nnn1C N1(C(c2cnn(C)n2)=O)CC2CC(NC(=O)C3=NOC(c4cnn(C)c4)C3)CC2C1 C1(C(N2C(C)CC(CNC(=O)Cn3cc(Cl)cn3)C2)=O)CCCC(=O)N1C N#Cc1ccnc(NC(C2CN(Cc3cccc(F)c3Br)CCC2O)=O)n1 n1(CC(=O)N(CCCNC(COCC(=C)C)=O)CCO)cnc(C(N)=O)n1 C1(C)(NC(=O)NCCC(COC)O)CCCC1OC N1(C(CC2N(C(COCCCOC)=O)CC(O)C2)=O)Cc2ccnn2CC1C N1(CC=C)CCC(C(N2CC3C(C(=O)NC4CC(CCC(N)=O)C4)C3C2)=O)CC1 C1(NC(CCSCC)=O)CC12CCN(C(=O)CC1(n3ccnc3)CC1)CC2 Cc1cc(=NC2CCCN(c3cnccn3)C2)[nH]c(N2CCOC(C)C2)n1 CC(C(=O)NCCN(C(c1ccn(C(C)(C)C)n1)=O)C1CC1)S(C)(=O)=O N1(C(C(CC=C)CC)=O)CC(C(=O)NCC(C)(C)C2CCCO2)CC(C)(C)C1 c1(C(N2CC(CC)C(NC(=O)Cc3cnc[nH]3)CC2)=O)ccc2nnn(C)c2c1 N1(C(c2ccnc(OC)c2F)=O)CC2CN(C(=O)CCCSC(C)(C)C)CC2C1 N1(C(c2cccc(SC)c2)=O)CCC(F)(F)C(C(N2CCC(C)(C#N)C2)=O)C1 N1(C(C2(COC)CC2)=O)CCC(CNC(C2C=CCCC2)=O)CC1 c1(CCN=C(NC(c2cccs2)C)NCCS(C)(=O)=O)cccc2ccccc12 C(=O)(C#CC1CCCO1)N1CC(CNC(c2oc(CC)c(C)c2)=O)OCCC1 C#CC1CCC(C(N2CCC(NC(c3[nH]c(C)nc3CC)=O)C(O)C2)=O)CC1 c1(C(N2CCCC(c3cn(CCN(S(C)(=O)=O)C)nn3)C2)=O)occ2c1CCC2 N1(C(C(F)=CCOC)=O)CCCCC(NC(=O)CCc2ccc(OC)cc2)C1 n1(CCOC)cc(C(=O)NCC(C)CN(C)C(c2csc(C(=O)OC)n2)=O)cn1 c1(C(=O)NCC2C(CNC(CNS(CC)(=O)=O)=O)C2)ccc2c(c1)NC(=O)CCC2 c1(OC)cc(C(N2CC(CNC(=O)C(C)C(F)F)C(C)C2)=O)cc(Cl)c1 C1(CC)CN(C(c2ccn(COC)n2)=O)CC1C(N1CCCC(CO)C1)=O c1(C2CCNC2)cccc(F)c1.O=C1NCCN1C1(c2cn(C3CC3)nn2)CC1 c1(Nc2ccc(C(=O)NC)cc2)cccc(F)c1F.c1(COC)nnnn1CCOC N(C)(S(=O)(=O)N1CCCCC1C)C(c1c(OC)nccc1)C#N C1(NC(c2cccc(CC)n2)=O)CC2CC1CN(C(=O)Cc1cnn(CC)c1)C2 Cc1n[nH]c(C)c1C(C)C(N1CCCC1CCCNC(=O)CCCCF)=O c1(NC(C2CC(C(=O)OCC)C23CCC3)=O)ccc2[nH]c3c(c2c1)CCCC3N N(C(=NCCC(=O)N(C)C)NCCCOCc1ccccc1)CCCC c1(CN2CCC(NC(c3n(C)cc(Br)n3)=O)C2)cc2ncccc2[nH]1 c1(C(N(CCNC(c2cc(C)c(CO)cn2)=O)C)=O)cc([N+](=O)[O-])c(O)cc1N C1(C(=O)NC2C3CCN(C(C(c4cccc(C)c4)=O)=O)C32)CCCC(C)(C)O1 c1(C(N(CCC(=O)NCc2c(C)scn2)CCO)=O)noc(C2CC2)c1C c1(C(=O)NC2CN(C(CCCCSC)=O)CC2C)cc(O)nc2ccccc12 C(C1=CCN(C(c2ccno2)=O)CC1)NC(C(Cc1ccccc1)NC(C)=O)=O C(=O)(C1=CCC2CCC1N2C(C12CCCC1C2(F)F)=O)N(CC#C)CC C1(C)(C(N2CC(C)C(Nc3ncc4ccnc-4[nH]3)C2)=O)CCCCNC1=O c1(C(N2CC(S(C)=O)C2)=O)ccc2c(c1)CCC2NC(C)(C)C c1(CC)cc(Cl)ccc1C(=O)NC(C1CCOC1)CNC(c1coc(O)n1)=O N1(C(C2(COC)CN(C(=O)COCc3nc[nH]n3)C2)=O)CCC(C)(OC)C1.C1CC1 C1(C(=O)NC(CNC(C(C)=C(CC)C)=O)C(C)(C)C)CC2(C1)CC21CC1 C1(NC(C=C(C)C)=O)CC2(CCCCN2C(=O)CSc2cccs2)C1 C1(C(=O)NCCN(C)CCO)(N(CC#N)C)CCC(F)(F)CC1.C(=O)(NC)N Cc1ccc(C)c(N(C(C2CCCN(C(=O)Cc3ccoc3)CC2)=O)C2CC2)c1 C1(NC(CC2(C(=C)F)CCC2)=O)C2CC1N(C(c1ccccc1C)=O)C2C C1(C#N)(CC(=O)NC(CNC(C(C)(O)C2CCC2)=O)C(C)(C)C)CCCCC1 c1(C(N(CCNC(C(n2ccc(C)n2)C)=O)C2CC2)=O)cnc2sc(C)nc2c1 Cc1nc(O)nc(O)c1NC(N1CCN(CC#Cc2cccnc2)CC1)=O N1(C(CCc2ccc(C)o2)=O)CCC2CC(NC(C3(C(F)F)CC3)=O)CCC2C1 N1(C(c2[nH]cc(CC)n2)=O)CCC(O)(C(C)NC(=O)C=C(C)Cl)C1 C(=O)(C1=NNC(=O)CC1)NCC(Cc1ccc(Cl)cc1)NC(CC#N)=O [N-]=[N+]=NC(CCC(N)=O)C(=O)NC1C=CCN(C(c2cc(C3CCC3)no2)=O)C1 C(CCC(O)C(=O)NCc1ccnc(O)c1)NC(CC1(CC)CCC1)=O n1(CCOC)cc(C(=O)N(C(C)CN(C(=O)C(C)NS(C)(=O)=O)C)C)cn1 C1(C(=O)NCc2c(C)csc2)CN(C(C2CCC(=O)N(C)C2)=O)C(C)(C)C1 CC1CC=CCC1C(N1CCC(CCNC(C2CN(C3CCOCC3)C2)=O)C1)=O N1(C(C(C)C2CCCC2)=O)CCC(NC(c2nnc(O)nc2O)=O)C(CO)CC1 C1(NC(C(COCC)NC(c2cc(C(N)=O)co2)=O)=O)CCC(=O)NC1C c1(C(N2CCC(C)(CCNC(C(CC)NC(N)=O)=O)C2)=O)cc(F)c(C)cc1N c1(C(N(CC(CO)(CO)NC(C2CCC(F)(F)C2)=O)C)=O)c(F)ccc(F)c1F C1(C(N(CC(CC)NC(=O)CC2(n3ccnc3)CC2)C)=O)CC=C(C)CC1 Cc1nc(O)[nH]c1C(=O)NC(CNC(=O)CN(c1cnccn1)C)CO C#CCC(C)(C(=O)N1OC2CCC1C2)NC(c1cc2n(n1)CCC2)=O N1(C(CN(CCOC)C)=O)CC(CNC(c2cc3occc3[nH]2)=O)C(C)(C)C1 C1(OC(c2cccc(-c3nn[nH]n3)c2)=O)CCCN(Cc2ccccc2Br)C1 C1(CCCC)C2=CC=NSC(CC)(CSC)CC(=O)NCCN(C(=O)C2)C1 c1(NC(N2CCC(C3N(C(CC(=C)C)=O)CCC3)C2)=O)cc2cccnn2n1 c1(C(=O)NCCOC2CCN(C(COC)=O)C2)cc(C)c(F)cc1F c1(C(=O)OC)cc2c(Br)c(NC(c3ncccc3F)=O)ccc2s1 Cc1nsc(C)c1C(=O)NCCCOCCNC(=O)C(C(C)C)NC(=O)C1CC1 N1(C(C(C(C)C)(F)CNC(C2(C)C=CCC2)=O)=O)CC2(CNC(=O)N2C)C1 N1(C(c2c(C)c(Cl)c(Cl)s2)=O)CCCC2(CC(NC(c3ccncn3)=O)C2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1CCCC(CCNC(c2nn(C)c(C#N)c2)=O)CC1 CN1CC(C(=O)NCC2(C)CCCN2C(c2cc(Br)no2)=O)NC1=O c1(C(=O)NCC2ON=C(C)C2)[nH]c2ccc(F)cc2c1Cl c1(C(=O)NC(CC)CNC(C2(C)CC(F)C2)=O)ccc(NC(C)=O)cc1C Cc1c[nH]c(C#N)nc1=NC(C)C1CCN(C(c2cn3c(n2)COCC3)=O)CC1 c1(C(=O)NCC(N2CCC(C)(c3ccccc3)CC2)=O)cc2cn[nH]c2cc1O c1(C(=O)NC2CC(C)(CNC(CSCC#C)=O)C2)cccn(CC)c1=O c1(C(=O)NC2CCN(C(CSCC#N)=O)C2)ccc(I)cc1 N1(C(C2CC2(F)F)=O)CCCN(C(c2cc(C(F)(F)F)n[nH]2)=O)C(CO)C1 c1(C(C(=O)NC(c2ccccc2)C)N(CC#CC)C2CC2)ccccc1Cl C1(F)(CNC(C(C)OCOC)=O)CCCN(C(c2cccc(C#N)c2)=O)C1 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(CCC(C)OC)=O)C(O)C(O)C1 CCC(CC)C(=O)NC1CCN(C(c2cc(OCC(F)F)ccn2)=O)CC1 C1(CNC(C2(C#C)CNC2)=O)CCCCN(C(=O)C(C)C(F)(F)F)C1 c1(C(N)=O)ccc(C(=O)NC2CCN(CCCNC(C3CC3C#N)=O)C2)cc1 C1(C(N2C(C)CCCC2)=O)COC2(CCN(Cc3cccc(O)n3)CC2)C1 c1(NC(C(n2ncc(NCc3ccc(C)s3)c2)C)=O)ccc2ncnn2c1 C1(=O)CCCCC(=O)N1.CC(C)CC(CNC(C1CCOC1)=O)N1CCOCC1 c1(C(=O)NC2C(SC)CN(C(=O)CSC(C)C)C2)ccc2nsnc2c1 c1(CC(C)N(CC)Cc2c(Cl)noc2C)ccc(Br)cc1 c1(CNC(C23CC2CN(CC2CC4C=CC2C4)C3)=O)ccccc1O Cc1cccc(Br)c1C(C(N1CCC(C(N)=O)C1)=O)NC(c1cccnc1O)=O C(CCC(=O)N=c1cc2ccccn2[nH]1)N(C)C(c1cccc(C)c1F)=O CN=c1nc(N2CC3CC2C2CC32)[nH]c(=NCC(C)(C)S(C)(=O)=O)[nH]1 c1(C(=O)NCC(C)NC(c2c(C)cc[nH]2)=O)cnn(C(C)C)c1Br C1(NC(Cc2ncc(C)o2)=O)CC(F)CN(C(c2ccc(-c3cc[nH]n3)s2)=O)C1 Cc1[nH]ccc1S(=O)(=O)N1CCC(F)(CNC(=O)N(C(C)(C)C)C(C)C)CC1 C1(C)(NC(C=CCNC(c2c(CC)nns2)=O)=O)CCC(C)=C(C)C1 C(CC(C(=O)N1CCC(CF)C1)NC(=O)COc1cnn(C)c1)=CC N1(C(Cc2ccn(C)c2)=O)CCN(C(C2(C)CC2c2ccccc2)=O)CC1 Cc1csc(=NCC(=O)NC2(CNC(C3CC4COCC4C3)=O)CCOC2)[nH]1 C1(C(N2C(CNC(C3C4CCN3CC4)=O)CC(C)(C)C2)=O)CN2CCCN1CC2 CCC(C(F)C(=O)O)NC(c1ccc(CN2CCOCC2)cc1)=O Cc1cnc(C(N2CCCCC2CNC(=O)CNS(=O)(=O)C2CC2)=O)cn1 C1(CNC(C2CC(OC)C2)=O)CCCCN(C(C2(C)CCCC2C)=O)C1 C1(C(=O)NC2C(C)CN(C)C2)C(C2CC2)CCN1C(c1ccccc1)=O N1(C(c2c(C)nccc2)=O)CC2CC1CN2C(c1cc(C(N)=O)[nH]n1)=O c1(N2CC3CN(C(COC)=O)CC3C2)ccc(S(=O)(=O)N2CCCC2)cn1 c1(C(C(=O)N(CCC)CCNC(=O)Cn2cncn2)n2cccc2)ccccc1 N1(C(C(CC)n2cncn2)=O)CCCN(C(=O)C(C)OC(C)=O)CC1C c1(-c2n(CC3C(C)OCC3)nc(-c3ccn(C)n3)n2)cnc2ccccn12 CCC(CC)CN=C(NCc1ccc(F)cc1)N1CC2C(C1)C2(C)C c1(NC(C(CC=C)C)=O)ccc(C(=O)NC2(C)CC2)cc1C c1(C(N2CCC(CCC(N)=O)C2)C(=O)NCCCSC)sccc1Cl C1(OC)(CNC(=O)C=CC(=O)NCC(N2CC(N3CCNC3=O)C2)=O)CCOC1 N1(C(C(CN(C)C)N(C)C)=O)C(CC(=O)N(C2CC3CC3C2)C)C2CCCC12 C(=O)(C(CCS(C)=O)N(C)C)N(CC(C)(C)NC(C1C(C(C)C)CCO1)=O)C C1(CNC(C(C)SC)=O)CC2(CCN(C(c3ccc(C)c(F)c3)=O)CC2)CO1 C1(C(=O)NCC2N(C(C3C(C(=O)OC)C3)=O)CC(C)(C)C2)CCC(C)C(C)C1 C1(CNC(Cn2c(C)nc(C)n2)=O)CC2(C1)CN(C(C1C=CCS1)=O)C2 c1(C(=O)NC2CC(CCNC(CN(C)CC)=O)C2)noc2c1CC(C)(C)CC2 C(=O)(CCCCCN(C(=O)C(N1CCOC1=O)C)C)NC1CN(CC)CC1C C1(NC(C2CCCN(C)C2)=O)CN(C(=O)CSc2nncs2)CC(F)(F)C1 CC(C)C(O)C(=O)NCC1CC(NC(c2ccn(C)c2)=O)C1 c1(CC(=O)N(C2CCN(C(=O)OC(C)(C)C)C2)CC)cc(C)nn1C c1(NC(C(c2ccc(F)c(C)c2F)N2CCC(SC)C2)=O)ccc2c(c1)OCO2 CCC(C)C(O)C(=O)NCC1CC(CN=c2[nH]ncs2)C12CCC2 c1(COCC(=O)NC(CC)CNC(C2CC(SC)C2)=O)cccnc1 N1(C(C(C)OCC#C)=O)CCC(C(=O)NCCN(C)CCF)C1 C(=O)(C1=CCCCO1)N1C2(C(=O)NCC3(CCOCC)CC3)CC2CC1 C1(C(C)C)CN(C(c2cccn2C)=O)CCCN1C(c1cc(C2CCC2)no1)=O C1(C)(CCC(=O)NC2CC(CC)C2)CCCN1C(=O)C(C)C(=O)OC c1(C(=O)NC2C(NC(=O)NC(=O)C(Cl)(Cl)Cl)C2)cc(F)cc(Cl)c1 c1(CC)ccc(Cl)c(C(N2CCN(C(C3CCCC3(C)C)=O)CC2C2CC2)=O)c1 C(S(C)(=O)=NC(=O)CCOCC1CCCC1)c1ccc(C)cc1 C(=O)(C(C)CCNC(=O)CC=C(Cl)Cl)OC.C12(CSC1)C(=O)N2 N1(C(c2c(CC)cco2)=O)CCC2CC(C(=O)NCCc3ccsc3)C2C1 c1(C(N(C2C3CN(C(CC(CC)C(F)F)=O)CC32)C)=O)ccc2oc(O)nc2c1 Cc1ccc(F)c(CC(=O)NCC2CC2CNC(C2OCCC2C)=O)c1 C1(CNC(CCN(c2ccccc2)C(C)=O)=O)CCN(C(=O)Cc2ccc(C)s2)C1 N1(CC)CC2CC1CN2C(=O)C(Cn1cccn1)NC(C12CC(C1)C2)=O Cc1[nH]c(C(C)(C)C)cc1C(N1CCN(C(C23CCC2C3)=O)CC1)=O C(CN=c1[nH]c2cccc(F)c2s1)C1N(C(C2C(C)(C(C)C)C2)=O)CCCC1C c1(C(=O)NCC(C)NC(C2(CCOCC)CCCC2)=O)coc2cccc(C)c12 C1(NC(C2(c3ccc(N(C)C)cc3)CC2)=O)CC2CC1N(C(=O)C(O)CF)C2 Cc1cc(C(N2CCCC2C(=O)NCCCNC(N)=O)=O)cc(O)n1 c1(C(=O)NC(C2CCCCC2)CNC(CCOC)=O)cnc(N2CCOCC2)s1 c1(CN(CCN(C(C(C2CCC2)OC)=O)C)C)cnn(C)c1-n1cnnc1 c1(C(=O)NC2CN(C(Cc3scc(C)c3)=O)CC3C2C3)cccc([N+](=O)[O-])c1 C1(NC(C(C(CC)C)OC)=O)CCN(C(C2(C(=O)N(C)C)CC2)=O)CCC1CO C#Cc1cccc(NCC[Si](C)(C)C)c1.C12CCN(CC1)CCCO2 n1(CC(=O)NCCCNC(C2CCC(C)(O)C2)=O)nnc2ccccc12 Cc1ccc(Cc2nc(-c3ccc(C)o3)nn2Cc2cccs2)c(Cl)c1 C(C(=O)Nc1cccc(C(=O)NCC2CC2C2CC2)c1)(C(C)C)NC(C)=O CCCCCCC(CC)C(=O)NCC1CCCN1C(c1ccc(C)[nH]1)=O c1(N(C)Cc2scc(C)n2)nc(NC2CCC(=O)NC2)c2ccsc2n1 C(=O)(C1CCC(=O)c2ccccc21)N1CCC(C)(CNC(=O)C=CC=C(Cl)Cl)C1 N1(C(C(C)=C(C)C)=O)CC=C(CCNC(C2CC2c2ccccc2)=O)CC1 C(=O)(C1=CCCC1P(C)(C)=O)NC(CC)CN(C)C(c1ccc(Cl)o1)=O C1(CC)CCCCC1N(C(=O)Cc1cccc(SC)c1)C.C12CCN(C1)C2=O C1(C(N2CCN(C(C(C)(C)OC(C)=O)=O)CC2)=O)CCn2c(cnc2C)C1 C(c1ccccc1F)=CCC(=O)NC12CN(C(C3(OC)CCC(C)C3)=O)C(C1)C2 c1(CC)c(C(=O)NCCCC(C)NC(=O)C(C)(F)CC)nnn1CC CCCS(=O)(=O)CC(=O)N1CC(C(C)NC(=O)CCc2ncccc2C)C1 N1(C(CCNC(N)=O)=O)CCCC1C(=O)NCCNC(C1(c2ccccc2)CC1)=O C(C)(C)(CC(=O)N1CC(COCCC(=O)N2CCC2)C(O)C1)OC Cc1nc2ccc(C(=O)NCCC(C)N(C(=O)CN(C)C3CC3)C)cc2[nH]1 C1(C)(C(N(C)CC2C(NC(C3CCC(C)CC3)=O)CCCC2)=O)CCOC(C)C1 C(C(=O)N=c1cc2ccccn2[nH]1)(N(C(=O)CP(C)(C)=O)C)C1CC1 c1(CNC(N2CCC(OC)C2)=O)cccc(S(=O)(=O)NC(C)(C)CC2CC2)c1 C1(CNC(=O)NCC2(c3c(OC)cccc3)CCCC2)CC(=O)C12CCC2 N1(C(CCSCCCC)=O)CC(C(=O)N(C)Cc2cccnc2)CC1(C)C C(CP(C)(C)=O)Nc1c(C(c2nnnn2C(C)(C)C)SC)scc1 N1(C(C2N(C(C(C(C)C)C)=O)C(C(C)C)CC2)=O)CC2CCC(C1)C(O)C2O C1(NC(Cc2cc(C)no2)=O)CC2CC1CN(C(=O)CCc1cnn(C)n1)C2 CC(=O)CCC(=O)NC(c1nocc1C(=O)NC1CCC2CC12)C N1(C(c2c(C)nco2)=O)CC2(CO)CC1(C(=O)NC(c1ccc(F)cc1)C)C2 c1(OCC)cc(F)cc(C=CCN2CCCC2c2ccnn2C(C)C)c1 Cc1nn2ncccc2c1C(N1CCC2CC2(NC(c2ccsn2)=O)CC1)=O N1(C(c2ccc(C#C)cc2)=O)CC2(CCC(C(N3C(C(N)=O)CCC3C)=O)O2)C1 CON(CCC(=O)N1CC(C)CCCC1C)C(=O)c1cnnn1C1CC1 CC(C)CC(F)C(=O)NCc1ccccc1-n1cc(CNS(N)(=O)=O)nn1 C(CC(C(=O)NOCc1ccccc1)NC(=O)C(C1CCOCC1)O)OC c1(C(N2C(C)CC(CNC(CN(C)C(=O)C3CC3)=O)C2)=O)cc2cc(Cl)sc2[nH]1 C(=O)(N=c1cc(-c2ccco2)o[nH]1)NC(CCC(F)(F)F)c1c(C)cccc1 c1(C(=O)OCC)nn(C)c(=O)cc1C.C1(=O)COCCOCCOCCN1.CCCO c1(SC)ncc(Cl)c(C(=O)NCC2(F)CCN(C(c3cccnn3)=O)C2)n1 C(=O)(n1[nH]c(=NC(=O)C2(C)CC2)c2c1CN(C(=O)C(C)(F)F)C2)OC C1(C(=O)NCC(F)CO)CCCC12CCN(Cc1ccc(O)c(I)c1)C2 C1(CNC(CC(=C)C)=O)CN(C(=O)Cc2ccc3n[nH]cc3c2)CCC1(C)C C(=O)(C(C)(C)CCC#N)NCC(CC(=O)NCC1CN(C(C)C)C1)C1CCC1 C1(CCC)CN(C(=O)C=Cc2cnn(C)c2)CCN1C(C1CC1(C)C(C)(C)C)=O c1(C(N2C3CN(Cc4cccc(O)n4)CC23)=O)c(Cl)cccc1I C1(C(=O)NC(C#N)C(N)=O)CC2(CC(NC(c3ccnc(Cl)c3Cl)=O)C2)C1 CC1CCN(C(=O)Cc2ccnc(F)c2F)CC1CNC(c1cnc(O)s1)=O C1(NC(CCNC(C)=O)=O)(CNC(C2CCCSC2)=O)CC2CCC1CC2 Cc1ccc(C(N2CCCC2C2(NC(c3ccnn3C(F)F)=O)CC2)=O)cc1N c1(NCCC=CC=C)[nH]c(=NCCC(C)(C)OCC)nc2c1ncn2CC S(=O)(=O)(c1ccc(CNC(N2CCn3cc(F)cc3C2)=O)cc1)NCC c1(CC)occ(C)c1C(=O)NCCCN(C(C1CC(F)C1)=O)C1CC1 N1(C(c2cn(C)nn2)=O)CCCC(c2cn(CCN3CC(CF)C3)nn2)C1 C1(NC(CN(C)CC)=O)CN(C(c2ncc(C)cc2C)=O)CC(C)(C)C1 N1(CC(=O)NCC2(CCNC(C(C)CC3CCC3)=O)CC2)C(C)CCC1C c1(C(=O)Nc2nccc(CNC(CN(C)CC)=O)c2)nc(CN)cc(O)n1 N1(C(CSCCC#N)=O)CC2CC(NC(=O)Cc3cc(Cl)ccc3Cl)CC1C2 c1(NC(c2nnnn2CCCF)(COC)C)ccc(S(C)(=O)=O)c(Cl)c1 c1(NC(CC)CNC(C2CCN(C)C2)=O)nc(C)cc(C)c1C(=O)OC C1(CC)C(NC(=O)CCc2cccnc2)CCN1C(c1coc(Cl)c1)=O N1(C(C2CC(C)(C)C2)=O)CCC(O)(CNC(c2ccc(CO)cc2)=O)C1 Cc1cnn(C)c1CC(=O)NCC(C)(C1CCC1)NC(=O)CC12COC(C)(C1)C2 c1(COC)cccc(C(=O)NC2CC(CNC(C3(C)C=CCCC3)=O)C2)n1 c1(CCC(=O)NCCCCSc2nn[nH]n2)ncc(-c2ccncc2)o1 N1(C(C(F)=C(C)C)=O)CC(NC(=O)CC2CCCOC2)C(N=[N+]=[N-])C1 Cc1cccc(C(C)NC(C2CN(S(=O)(=O)Cc3cncnc3C)CCN2)=O)c1 C(=O)(CCCCC(C)(C)C)N1CC(C2(NC(Cc3n(C)ccn3)=O)CC2)C1 N1(C(C)(C)C)CC2C3C=CC(C3)C2C1.N(C)(S(=O)(=O)NCC=O)c1scc(C)n1 c1(C(N(CCCCCC)CCNC(=O)C(C)CSC)=O)nc(Cl)c(CC)[nH]1 N1(C(Cc2cccc(SCC)c2)=O)CCN(C(=O)CC2CCSC2)CC1CO N(C1COc2ccc(Br)cc21)N1C(=O)OC(c2ccc(OCC(F)F)cc2)C1 C1(CC(=O)N(C2CCN(C(C(CC)SC)=O)C2)CC2CC2)CC2(CCC2)C1 c1(CNC(C2CC(F)C2)=O)nc2c(s1)CCN(C(=O)CCCF)C2 CC1(C)CC(C(=O)NCC2CN(CCF)C2)CN1C(c1cc(C(F)F)no1)=O c1(CC2(C(N(C3CN(C(C4CCCO4)=O)C3)C)=O)CC2)ccccc1 c1(N2CCCC(CCNC(=O)C=CCO)C2)ccc([N+](=O)[O-])cn1 C(=O)(C(C(C)(C)O)NC(=O)C=CC1(C)COC1)N1CCC(CSC)C1 c1(C(=O)NC2(C)CCN(C(c3cnc(C(C)(C)C)o3)=O)C2)cccc2cncn12 N1(Cc2n(C)ncc2-c2cnsc2)C(C2CC2)CC2CCCC12 C#CCC(CC(F)F)C(=O)NC1COCC1NC(=O)C(C)SCCCC Cc1csc2c(C(N3CC(CC(=O)NC(c4ccc(Br)cn4)C)C3)=O)ncnc12 c1(C(=O)NCC2C3CN(C(c4c(C)cccc4)=O)CC32)cccc2c1OCC2C c1(C(=O)NCC(C)NC(c2ccnn2CCN(C)C)=O)cnn(C)c1Cl c1(C(c2nnnn2CCCF)(C)NC2CCC2(C)C)ccc(F)cc1Br N1(C(COCCOCC#C)=O)CCCC(F)(NC(c2ccc(OCC)nc2)=O)C1 CCCC(C)CC(=O)N1CC(O)(C(F)C(=O)NC(CCO)C(F)(F)F)C1 C1(NC(c2c(OC)scc2)=O)CC2(C1)CC(CNC(C1(C)CC1(F)F)=O)C2 C(=O)(CC(C(F)(F)F)OC)N1CC2(CN(C(c3cc(CC)no3)=O)C2)C1 C#CCC(C(=O)NCCCOCC)NC(c1cc[nH]n1)=O C1(C(N(C(CNC(=O)CC(C)F)C2CC2)C)=O)CC(=O)N(C(C)(C)C)C1 Cc1ccc(C(=O)NC2CC(O)CN(C(=O)Cn3cccc3)C2)cc1S(N)(=O)=O C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(CC=C)NC(=O)CN(C(=O)COC)C c1(C(=O)NC(CC(C)NC(=O)Cc2cnn(C)n2)C)c(Cl)cnn1C Cc1c(C(=O)NCCC2=CCN(C(C3CC3F)=O)CC2)[nH]c2c(Cl)cccc12 C1(C(N2C(CCNC(C3(C)CCOC3)=O)CCC2)=O)CC2C=CC1C21CC1 C1(NC(Cc2c(C)occ2)=O)CC2CCC1N(C(c1c(C)n[nH]c1C)=O)C2 c1(C(C)C)cc(C(N2CCOC(CNC(C3(N(C)C)CC3)=O)C2)=O)cc(Br)c1 N1(C(C(CCSC)NC(c2ccc(C#N)cc2)=O)=O)CC(C)CCCC1C c1(CNC2C(C(=O)Nc3c(C(=O)OC)c[nH]n3)C2)cccc2c1CCCC2 C(CC1=CCN(C(=O)C(C)n2cnnn2)CC1)NC(C(c1cccc(F)c1)C)=O C(CNC(c1cn(C)c(=O)n1C)=O)(CC(F)(F)F)NC(Cc1ncc(CC)[nH]1)=O C(C1(O)CCc2ccccc21)NC(=NCCC)N(C)CC(c1ccsc1)OC CCC(F)(C(=O)OC)C(=O)N1CC(N(C(=O)Cc2csc(S)n2)C)C(C)(C)C1 C(=O)(C(F)(F)C(F)(F)F)N1CCN(C(CC2CC(C(C)(C)C)C2)=O)CC1 CC12CCC(C)(O1)C(C(=O)N(C1CCNCC1)Cc1ccc(Cl)cc1)C2 c1(-c2nc(C3CC(C)(C)SC3)on2)ccc2c(c1)OCC2 C12CCN(CC1C1CC1)C(=O)N2.C=Cn1nncc1C(NOC(=O)OC(C)(C)C)=O N1(C(COCC#C)=O)CC(NC(=O)C(C)(O)CCC)CC2(CCC2)C1 c1(OC)cc(F)c(F)cc1C(=O)NC(C)C(C)NC(=O)CSCC(=O)OC c1(NC(c2n(CC)nnn2)C(C)(C2CCOCC2)OCC)cccc(OC)c1 CCCCCCCCC(=O)N(CC(C)CNC(c1cnn(C(C)C)c1C)=O)C c1(CC)nc(C(c2nnnn2CC)NCC(N2CCCC2)C)cs1 CC1(OCC(=O)NC(C(=O)NCc2cncn2C2CC2)C2CCOC2)CCCC1 C1(NC(C=Cc2ccc(C)s2)=O)CN(C(=O)Cc2ccon2)CC12CCC2 C(=O)(CS(C)(=O)=O)OC.CCC(C)N1CC1 c12cc(ccc1Br)C(=O)Nc1ccc(cn1)C(=O)N2.N1(CC)CCOC(C#N)C1 C1(CNC(C2C(=C)CC2)=O)CN(C(=O)CC2(O)CCCOC2)CCN1C c1(NCCCCSC)nc(N2CCC(CC#N)C2)nc2scnc12 C1(C(N2C(CCNC(Cc3nc(COC)sc3)=O)CCC2)=O)CCS(=O)(=O)N1 N1(C(C(=O)NCC)=O)CC(NC(c2cccc3c2NCC3)=O)CC12CCOCC2 C1(NC(CC(=C)C)=O)CCC2(CC1)CC(CNC(=O)C(=O)NCCCC)C2 N1(CC(C2CCC2)C(=O)OC(C)(C)C)CCCC(C(N)=O)C1 c1(CCNC(=O)NC2CCC2)ncn2c1COCC2 C1(CNC(C=CC)=O)CCN(C(c2ccc(C(F)F)nc2)=O)CC1(F)F C1(C(=O)NCC(n2c(C)nc(C)n2)C)CN(c2ncccc2C(=O)O)CCN1C c12ccc(c(F)c1)S(=O)(=O)N2.C1(C)CN(c2ccc(C(=O)N(C)C)cn2)CCN1 N1(C(C(C)=CCC)=O)CCC(C)(C(N2CCC2C=C)=O)CC1 c1(C(=O)NCCC(=O)NCC2CCC(C(C)C)CC2)cc2n(n1)CCC2 N1(C(Cc2cc(CC)no2)=O)CC2CCCC1C2CNC(C1CCCO1)=O CCCS(=O)(=O)C(C)C(=O)N1CC(OC)CC(NC(=O)Cc2ccc(C)nc2)C1 CC1(C)CCN(C(=O)CCC2CC2)CC1.c1(C(=O)NC=O)nccc(O)n1 N1(C(CC2N(C(C(C)OCC=C)=O)CC2)=O)CCN(C(C2CCC2)=O)CC1 CCCC(C)C(=O)NC1(CCNC(=O)CSc2nncn2C2CC2)CCC1 N1(C(c2cncc(NC)c2)=O)CCC2(NC(c3cnc(C)cn3)=O)CC2C1 C(=O)(C(C)(O)CC(F)(F)F)N1CCC(CNC(C(C)(C)N(S(C)(=O)=O)C)=O)CC1 C(=O)(CC(C)C(F)F)N(C1CCN(C(c2c[nH]nc2Cl)=O)CC1)CC c1(CC)nnc2n1CCCC2C(=O)N1CCC(N(C(=O)CC2CCC2)CCO)C1 c1(CC(N2CCC(N(C(C(C)CC3CC3)=O)C)C2)=O)ccc(O)cn1 NS(=O)(=O)CC(=O)NCc1cn(CCNC(C2CCOC2C(F)F)=O)nn1 N1(C(c2c(C)cnnc2)=O)CCCC(C)(C)C1C(=O)NCC(c1ccncc1)C C1(NC(c2c(CC)nns2)=O)CCCC2CN(C(=O)Cn3cc(C#N)cn3)CC12 C(=O)(C1=CCCOCC1)N(C(CNC(=O)C1=CSCCO1)C1CC1)C C1(NC(=O)C=CCO)CN(C(c2cccn2Cc2ccccc2)=O)CCC1CO N1(C(C2C(=C)C2)=O)CCOCC(CNC(c2cc(-c3ccc(F)cc3)no2)=O)C1 Cc1cccc(CNC(C2C3CC2N(C(=O)C=Cc2cccc(O)c2)C3)=O)c1F C1(C(N(CC(C)CNC(C2(C)C=CCC2)=O)C)=O)CC(=O)CC(=O)C1 c1(CC(=O)N(C)CC2(NC(c3ccn(CO)n3)=O)CC2)cnc(-c2cccs2)[nH]1 C(C)(C(=O)NC1CC2(C1)CC2NC(c1ccc(Cl)c(N)c1)=O)(C(C)C)NC(C)=O C1(C2(O)CCN(N(CC3CCOC3)CC(C)C)CC2)(C(=O)OC)CCOCC1 c1(OC)cccc2c1CC(CC(=O)NCc1ccc(N3CCCC3=O)cn1)C2 CCCCCC(=O)NCC1C(C)CCN1C(=O)CC12CC(c3ccccc3)(C1)C2 C1(CNC(CSCC#C)=O)CN(C(=O)C#CC2CCCCO2)C2(CCOCC2)C1 c1(OC)ccc(N)c(C(=O)NC2CCN(C(c3cc(Cl)cs3)=O)C2C)c1 c1(C(C)C)ccc(C(=O)NCC2CC(O)CN2C(=O)CCC(F)F)cc1F C12(NC(=O)NCCCN3CCC(OCC)CC3)CC(CSC)(CCO1)C2 c1(NC(=O)NC2CCN(CCC(=O)OC)C2=O)cc(Br)c(C)cc1F c1(NC(C(c2ccco2)NC(c2c(C)occ2)=O)=O)cccc(C(C)F)c1 C1(OC(C)C(=O)NC2CC2CNC(=O)CC(C)(C)C)CCOCC1 C1(COC)CN(C(c2cc(C)nn2C)C(=O)N(CCC2(C)CC2)C2CC2)C1(C)C CC1(C)CC2(CC(C(=O)NC3(C)CN(C(=O)Nc4ccc5c(c4)CCO5)C3)C2)C1 c1(C(N2C(CC)CN(C(C3CSC3)=O)CC2)=O)ccc2c(n1)OCCO2 c1(C(C)C)ncncc1C(=O)N(CC(C)(C)CNC(c1ccncc1)=O)C O=NN1CCCC1C(=O)NC1CCC(NC(=O)CC2CC(F)(F)C2)C1 C(=O)(C#Cc1ccc(O)cc1)N1CCCC(c2c(C)n[nH]c2C)C1 N1(C(c2ccc(C(N)=O)cn2)=O)CCC2(CC1)CCN(C(=O)CCOC1CC1)C2 N1(C(CS(CCOC)(=O)=O)=O)CCOC2CN(C(=O)Cc3nonc3C)CC12 CCCCC(C)C(=O)NC(C(=O)N(C1(COC)CC1)C)C1CCC1 C1(C)(NC(c2ccn(CC)n2)=O)CCN(C(C2CCC(C(=O)OC)C2)=O)C1 CC1(C)CC(C(=O)NCc2nnc(O)o2)CN(C(C2C3CCCOC23)=O)C1 c1(C(N2CC(C(=O)CCc3ccc(CO)[nH]3)C2)=O)ccsc1CNC(=O)OC C1(C(N(C(C)CN(C)C(c2cn(C3CCCCC3)nn2)=O)C)=O)CC2(C1)CC2F C(=O)(C1CCCn2nccc21)N1C(CNC(c2c(SC)cccc2)=O)CC(O)C1 Cc1ccc(C(N2CCN(C(=O)CCCCN(C)C)CC2C)=O)c(N)n1 C1(C(=O)NC(C(=O)N(CC(CC)OC)C)c2ccoc2)CC2(C1)CC21CC1 C(=O)(C(COC)NC(=O)Cc1ccsc1)NC1CC(CC(=O)OC)C1 c1(NC(C)(C)C)ccc(Cl)cc1CC(c1nnnn1C1(C)CC1)C1CCO1 CCC(C)(F)C(=O)N1CCCC(CN(C)C(c2ccn(C)c2C)=O)C1 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(C)(C)C(NC(c2nc(Cl)cs2)=O)CC1 C1(NC(CSCCCC)=O)CN(C(c2ccc(C(C)F)cc2)=O)CC1SC C1(C(N(CC(C)O)CCNC(c2ncc(OCC)nc2)=O)=O)CC2OC1C1CC21 C1(C(=O)NC23CC(C(=O)NC(CC(=O)NC)(C)C)(C2)C3)CCCCC(=O)N1 c1(OCCC)c(NC(=O)NCC2(C)CCCC(=O)N2)cccc1C C(=O)(CCCC(CC)NC(=O)CC(C)F)N(CCOCC=C)C c1(C(=O)NC2C(NC(C(CCSC)O)=O)CCC2)ccnc2[nH]ncc12 C1(CC(=O)NCC(C#C)C(C)C)CC(C)(C)CN1C(C1CC(=O)N(C)C1)=O C1(NC(c2cc(C)c(=O)n(C)c2)=O)CCC(N=c2[nH]c3ccc(F)cc3o2)C1 Cc1nc2cc(C(=O)NC3CN(C(=O)C(C)S(N)(=O)=O)CC3N=[N+]=[N-])cnc2[nH]1 N1(CC)C(=O)CCC1CC(=O)NC1CCC1NC(=O)CCCn1ccccc1=O c1(C(N2CCC(C)=C(Br)C2)C(=O)NC(CCSCC)OC)cc(Cl)cc(Cl)c1Br C1(NC(c2ncc(C)c(Cl)c2)=O)COC2(C1)CN(C(c1cc([N+](=O)[O-])sn1)=O)C2 CC1CC2(CCN(c3nnc(C4CC4)o3)CC2)CN1C(C1CC12CC2)=O Cc1ccnnc1C(=O)NCC(C(C)(C)C)NC(c1ccc(F)o1)=O C1(C(N(OC)Cc2ccc(C)o2)=O)CN(C(c2c(C)noc2N)=O)CC12CC2 Cc1ccc(CN(C(=O)C=CC(C)NC(C2CCCN(C)C2)=O)C)cc1 C(=O)(C(C)(COC)CC)NCC1CCCN(C(c2cnn(CCOC)c2C)=O)C1 C1(C(C)C)CN(C(=O)CC2CC3C=CC2CC3)CCCN1C(=O)C1=COCC1 C1(C(=O)NC2(C)CC(NC(c3ccc(Br)cc3F)=O)C2)CC2CCCC2C1 CC1(NC(=O)CCCC#N)CCN(C(c2cc(C(C)(C)C)no2)=O)CC1 c1(C(=O)OC)cc(C)cnc1NC1CC(NC(c2cc(O)nc(C)n2)=O)C1(C)C c1(C(N(CC(C)(C)C(=O)N(CCCCO)C2CC2)C)=O)cncn(C)c1=O C1(N)CCC2(CCCC2)C1.C(=O)(C(F)C(C)(F)F)C(C(CN)N(C)C)=O Cc1cc(C(=O)NC2CCC(N(C)C(c3cc(C4CCC4)[nH]n3)=O)CC2)n(C)n1 N1(C(C2(CNC(C3N(C(C)C)C(=O)CC3)=O)CCC2)=O)CC2(CO)CCC1CC2 C(=O)(C1=NN2CCCN=C2N1)N1C(CNC(CC(=O)NC)=O)C(C2CC2)CC1 n1(CC)ncn(NC(=O)C(F)(CNC(=O)CN(C)C(=O)OC)C(C)C)c1=O N(C(=NCC(C)(C)C#N)NC1COC1)CC(c1cccc(Cl)c1)N(C)C c1(OCC)cnc(C(N2CC(O)(C(F)C(=O)NCCNC(=O)CC)C2)=O)cn1 c1(C(c2n(CCCCC)nnn2)Nc2cnn(CCSC)c2)ccc(Cl)c(F)c1 CC1C(CO)NC(=O)C2(CC2)NC(=O)C(=O)N1.c1(C(C)NC2CC2)ccccc1 c1(SCC(=O)NCC(O)CNC(c2cnn[nH]2)=O)ccncc1F c1(C(=O)NC(CNC(C(CC(C)C)F)=O)(C)CC(C)C)cc2cc(O)ccc2[nH]1 N1(C(c2c(CNC(CC3CC(=O)OC3)=O)ccs2)=O)CC2C=CC1CC2 C(CCCCC(=O)N1CCCCCC1CCO)NC(=O)C=Cc1cnccn1 C(=O)(C(CC(C)C)C(N)=O)NCC(C1CC1)NC(CSCc1c(C)noc1C)=O C#CCCCCCC(=O)NC1CCCC(CC(=O)NC(C)CSC(F)F)C1 C(=O)(C1=CC(C)(C)C1)NCC1C(NC(c2cn(CC)nc2)=O)CCCC1 CCCCC(O)CC(=O)NN1CC(C)C(O)C(C)C1.c12ccc(cc1)C(=O)NC2 Cc1cc(N)c(C(=O)NCC(C)(C)CNC(c2cc3sc(C)cc3s2)=O)cc1F c1(C(CN(C(C2CCS(=O)(=O)C2)=O)CC)OC)ccc(F)c(Cl)c1 N1(C(c2cc(CC)nn2C)=O)CCCC(C(=O)Nc2cccnc2)CC1 CC1CN(C(c2ccc(OC(F)F)nc2)=O)CCN1C(=O)CCc1cc[nH]n1 C(=O)(C1=CCCCC1)N1CC(C(C(=O)NCC(C(N)=O)O)O)C1 c1(C(N2CCC(CSC)C2)=O)cc[nH]c(=N)n1.C1(=O)C(Cc2ccco2)N1.C(C)(=O)N c1(C(C(=O)NCC2CCCO2)N(C2CC23CCC3)C)nc2ccc(Br)cc2s1 N1(C(C2(NC)CCCC2)=O)CCC2CC2(C(=O)NC)CC1.N12CCC1(C)C2=O Cc1cscc1C(N1CCC1(C)CC(=O)NC1(C(C)C)CCC1)=O c1(C(N2CC(C)(C(N3CCN(C)CC3CO)=O)C2)=O)ccc2c(c1)c(I)nn2C Cc1cc(C(=O)NC2CN(C(=O)Cc3nc(C4CC4)cs3)CC2C)nc(C)c1 N1(C(C(=O)NCCC)Cc2ccccc2F)CCN(C(=O)OC(C)(C)C)CC1C c1(C(=O)NCC(CNC(c2c(C#C)c[nH]n2)=O)CO)cc2ccc(Br)cn2c1 c1(C(CC)NC(C)C(=O)Nc2ccc(C)cc2C(F)(F)F)c(OC)cccc1O C#Cc1cc(C(=O)NC2(CNC(C3(C#N)CCC3)=O)CCCCCC2)cc(F)c1 N1(C(C2(COC)C=CCC2)=O)CC2CCC1CN2C(=O)C(=O)Nc1ccccc1 CC1COC2(C1)CN(C(C1CCC3(CC3)N1C(C1(C)CC1(C)C)=O)=O)C2 c1(CSCC)ccccc1C(=O)NCC1(O)CN(C(=O)CC(C)N(C)C)C1 c1(CC(N2CC(C)(CNC(C3C(OC)CC3)=O)C2)=O)cc(Cl)n(C)n1 C12(NC(C(CC#C)C)=O)CCC(CNC(c3ccncc3F)=O)(C1)OC2 N1(C(c2cnn(C)c2F)=O)CCC(C2CC2NC(C2CCSC2)=O)CC1 Cc1cc(C(=O)NC2CCCC(NC(=O)C=CCCC(C)C)C2)cc(Br)c1 c1(N(CC(F)(F)CO)C(=O)OC(CCOCCOC)=O)ccccc1 N1(C(CC(=O)OCC)=O)CC2C(CNC(=O)CCSc3ccc(O)cc3)C2C1 CCCC(C#N)C(=O)NC(Cc1ccco1)C(=O)NC(c1ccnc(F)c1)C c1(SCC(=O)NC(ONC(=N)CN2CCOCC2)C)cccc(Br)c1 C1(NC(=O)NCCC2CCOC2)CCCCC12CC2 Cc1cc(NCC(C)NC(C2(C)CCN(C)CC2)=O)n2nc(C)nc2n1 C1(CCC)CN(C(c2cc(O)nn2C)=O)CCN1C(C1CC1c1ccnn1C)=O N1(C(C2CC(C(C3CC3)NC(=O)CCc3cn[nH]c3)C2)=O)C(CO)CC1CO C(=O)(C(CN1CCCC1)CCCN)NC(c1ccc(CC)cc1)COC C1(NC(C=CC2(C)CCOCC2)=O)C2CCCN(C(=O)CC3(C)CC3)C2C1(C)C C1(N(C(CSC)=O)C)CN(C(=O)Cc2ccc(-n3cnnc3)cc2)CC1F C1(C(=O)NC2C3CC2N(C(=O)CCF)C3)COC2(CCC2)C1 C(=O)(C1CCCc2c(Br)cccc21)NCCCN(C(C(C)NC(C)=O)=O)C C1(C2(COC(c3cn(CO)nn3)=O)CC2)COC(COCCOc2ccccc2)C1 CC(C)(C)CC(O)C(=O)N1CC(CNC(=O)Cc2ccc(Cl)s2)C(F)(F)C1 Cc1cnc(C#N)c(-c2csc(C(=O)NCc3ccoc3)c2)c1 C1(C(=O)NCCCNC(Cc2n[nH]c(=NC)s2)=O)CCN2CCOCC12 c1(C(=O)NCC2C3CN(C(C4(C#N)CCCC4)=O)C2C3)cc2c(F)cccc2s1 C1(SCC)CCC(C(N2CC(N3CCN(C(=O)C(=O)N(C)C)CC3)C2)=O)CC1 C(C)(C)(CC(=O)NCC(O)C(F)(F)F)NC(CC1(OC)CCC1)=O Cc1ncc(Cl)c(C(=O)NCC2(O)CCN(C(=O)CC3CCCC(C)C3)CC2)n1 C1(NC(CC(C)(O)C2CC2)=O)CCCCC12CCCN(c1ccc(C#N)nn1)C2 CCC(C(=O)N(C1CCN(C(c2cc(CO)on2)=O)CC1)C)C(F)(F)F c1(C(C(=O)OCC)(C)F)ccc(F)cc1.C1CCCN(C)C(=O)N1C.C(C)(C)(C)O C(=O)(CC(C)(C)C#N)N1CC(C(=O)NC(COC)C(=O)OC)C1 C#CCC(O)C(=O)NCCC1(O)CCN(C(c2ccn(CC)c2C)=O)C1 N1(C(C=NOC)=O)CCC(NC(=O)C=Cc2sccc2Br)C(F)C1 C1(NC(N(CC(C)C#N)CC)=O)COCC1OC CCCC(CC)C(=O)NC1(C(=O)NC(CC)CC(C)CO)CC1 S(=O)(=O)(CCNC(c1nnnn1CCCF)(CC)C1CC(F)(F)C1)NCC c1(OC)ccc(COC(=O)C(N2CCC(OC3CC34CC4(F)F)CC2)=O)cc1 c1(C(=O)NC2CC(NC(=O)C(F)CC3CCCC3)C(O)C2)ccc([N+](=O)[O-])s1 CCCC(C(=O)N1CCC2C(C(N3CCC(NC(=O)NC)C3)=O)C2C1)C(C)C c1(COC)ncc(C(=O)N(C)CCNC(C2(C(F)F)CCC2)=O)s1 CCC(C)(CC)C(=O)N1CCC(CO)(CNC(=O)C(C(C)C)NC(N)=O)CC1 Cc1ccc2c(c1)CC(C(N1CCN(C(c3ccnc(C)c3)=O)CC1CF)=O)S2 C(=O)(C(=O)C(C)(C)C)NC(C1CN(C(c2cnn(C(F)(F)F)c2)=O)CCO1)C Cn1cc(C#N)cc1C(N1CCC2C(NC(=O)Cc3cn[nH]c3)C2C1)=O C(=O)(C(C)CC(C)(C)C)NC(CN(C(c1cccc(OCC=C(C)C)c1)=O)C)C N1(C(c2cc(=N)[nH]cc2)=O)CCC2(CC1)OCCCC2NC(=O)CSC(F)F c1(C(=O)NC2CC(C)N(C(c3cn(C)[nH]c3=N)=O)CC2)c[nH]c2ccccc12 CC1(C)C(C(=O)NC2CC3CC(NC(c4ccc(C#N)cn4)=O)C2C3)CC1(F)F N#Cc1ccc(C(N2CCC(F)(F)C(CNC(=O)Cc3cn[nH]c3)C2)=O)c(O)c1 C1(C(N(CC(=C)C)CC)=O)CN(C(=O)COCC(C)(C)C)CCN1C C1(C(=O)NC(C(C2(O)COC2)=O)=O)CCCN(C(=O)C2CC2)C1.CC(CN)CN(C)C c1(C(N2CC(O)CC(NC(C3CS(=O)(=O)C3)=O)C2)=O)ccc2ncsc2c1 C1(CC=C)(NC(=O)CC(C)(C)O)CCN(C(C2CCC2(F)F)=O)CC1 C(=O)(C(C)(F)C(F)(F)F)N1CCC(C)(CNC(c2ncc(C)cc2C)=O)C1 C1(NC(=O)NCC(c2cccnc2)N(CCOC)C)CC(F)(F)C1C C1(CC)CCN(C(=O)C(C)CCOC)C1C(=O)NCCN(CC(F)F)C N=c1nc2nc(C(=O)NCc3ccc(-n4cnnn4)cc3)ccn2[nH]1 N1(C(C2C(=C)C2C(=O)OC)=O)CCC2(CC1)CC2CNC(C1CC1c1cn[nH]c1)=O C1(NC(C(N2CCOC2=O)C)=O)CC(C)(NC(=O)Cc2csc(S)n2)C1 c1(C(N2CCC(O)(CNC(CC)=O)C2)=O)cnc2ccc(Cl)cn2c1=O N1(C(CC=C(C)C)=O)CC(C)CCC1CNC(=O)COc1ccc(CC#N)cc1 c1(CNC(C2C=CC(CNC(=O)C(O)Cc3cnc[nH]3)C2)=O)ncccc1O C12(C(N(C)CC3CCCN3C(c3n[nH]c4c3CCC4)=O)=O)CC3CC(CC1C3)C2 c1(C(=O)N(CCCNC(C2(Cl)CC23CCC3)=O)C2CC2)cc2c(s1)CCOC2 CCC(C)CCC(=O)N1CCOCC(NC(=O)CCNC(=O)CC(C)C)C1 N1(C(CC2(OC)CCC2)=O)CC(CNC(=O)C=CC2CCCN2C)OC(C)(C)C1 C12(C(=O)NCCN(CC(F)F)C)CC(C)(CN1C(C1CC1[N+](=O)[O-])=O)C2 CC(C)(CC(F)F)C(=O)NCCSCc1cn(Cc2ccccn2)nn1 Cc1cc(CNCCNc2cc(N)n(C)n2)ncn1 C1(NC(CN(S(C)(=O)=O)C)=O)CCC(F)(CNC(=O)CCc2ccc(O)nn2)C1 CCCCCCC(=O)NCCC1(NC(C2CCN(OC)CC2)=O)CCCC1 C1(NC(C23C(C)(C)OCC2C3)=O)CC12CCN(C(=O)CC1CCC1)CC2 N1(C(CC2(C(=C)F)CCC2)=O)CC2(CCC2NC(c2cncc(C=C)c2)=O)C1 C=CCC(CNC(c1cc(Cl)cn1C)=O)C(=O)NOCc1ccccc1F N1(C(c2c(C#N)csc2)=O)CCC2(CC1)CC(CNC(=O)CCOCC(F)F)C2 C12(C(N3CCN(C4CCN(CC=C)C4)CC3)=O)CCC(F)C1CC2 C1(NC(c2ccnc(O)c2F)=O)CC2CC(NC(C3CC4C(C3)C4(F)F)=O)C1C2 N1(C(CC2N(C(C)=O)CCC2)=O)CCCN(C(C2CC=CC2)=O)CC1 CCC(CCc1ccccc1)C(=O)NC(C)CN(C(=O)C(C)CCO)C c1(C(=O)NC2(CCNC(C(C3CCOC3)OC)=O)CCC2)ccnc(CO)c1 N1(C(CCSCC)=O)CC2CC(NC(=O)Cc3c(C)nn(C)c3C)CC2C1 N(C1CCCc2n[nH]cc21)C(CC(CC#C)NC(C1CCC(=O)N(C)C1)=O)=O C1(NC(Cc2c(C)ocn2)=O)CC(N=c2[nH]nc(C(C)C)o2)C1(C)C c1(CCC(=O)N(C2CCCC2)CCNC(C2(CC)CCOC2)=O)ccc(Cl)nc1 C1(NC(=O)Cn2ccnn2)CC2CC(NC(C3CC3[N+](=O)[O-])=O)C1C2 O=C(N=c1[nH]onc1C1CC1)C1CCN(C(c2ccc(C(F)(F)F)nc2)=O)CC1 Cc1nn(C)cc1CNC(C1CCCC1NC(=O)CC=C(Cl)Cl)=O c1(OC)c(C(N2CCC(n3cncn3)CC2)C(=O)NCCCF)cc(C)cc1C c1(OC)cc(F)c(C(N2CCC(C(N3CCOC(=O)C3)=O)C(O)C2)=O)c(F)c1 C=CCC(C(=O)NC(CC(=O)N(CCC(C)C)C)C1CC1)NC(C)=O C1(C)(C(N2CC(NC(CSC(C)C)=O)C(C(F)F)C2)=O)CCC12CCC2 c1(NC(C2CCC(NC(c3ccc(F)cc3I)=O)CC2)=O)nccc(Br)c1Cl C#Cc1ccc(C(=O)NCC2CCCC(NC(=O)C(C)S(N)(=O)=O)C2)nc1 C1(SCC)CCC(c2nc(-c3ccn(C)n3)nn2Cc2ccsc2)CC1 c1(N2CCC(CC(=O)Nc3cc(OCC)ncc3)C2)nc(C)nc2c1CCC2 c1(C(=O)NC2C3CN(C(c4n(CCC)ccc4)=O)C2C3)cc2cccnn2c1 c1(NC(=O)C(C)(C)C)ccc(F)cc1.Cn1ccnc1C(=O)NCC1C(=O)O1 CC1(C)CC(CNC(c2sccc2F)=O)N(C(=O)C(O)C(F)F)C1 N1(C(C(c2ccc(F)c(Cl)c2)C)=O)CC(NC(c2cccnc2F)=O)CC1(C)C CC(C(=O)NC1(CNC(=O)C(C)N(C)C)CCC(C)(C)CC1)C(F)(F)C(F)F C(=O)(CCCCCc1ccc(OC)cc1)NCC(C)(C)NC(C=CC=CCC)=O C(=O)(C(O)CC(C)(C)C)N1CC(OCCNC(c2n(CC)cnn2)=O)C1 c1(SC)nc(NC2CN(C(=O)C3=CCCC3)CC2(C)C)ncc1C CC1(C(N2CCC(C(C)(O)CNC(=O)CC3CCSC3)CC2)=O)CCNC1=O N1(C(c2n(CC)nnc2)=O)CC(CNC(C2(SC)CC2)=O)CC12CCC2 N1(CC(=O)NCC2N(C(c3c[nH]c(=NC)o3)=O)CC=C2)CCC(=O)NC1=O C#CCC(C)(C)C(=O)N(C)CCN(C(=O)C(F)C1CCCC1)C c1(NC(=O)NCCc2cccc(C(=O)OC)n2)ccc2c(c1)ncn2C(C)C C1(CCC)CCC(N(C2CCCC2)C(=O)NCc2nc(C3CC3)cs2)CC1 c1(C(=O)NC(CC(C)NC(c2nc(CCC)sc2)=O)C)cnn(CCC)c1C S(=O)(=O)(CCCC1CC1)NC(=O)C(CN1CCCC1)c1ccccc1 C1(NC(CC(C)n2ccnc2)=O)CCC(F)(CNC(c2nc(C3CC3)cs2)=O)C1 C(=O)(C(CC(C)C)n1ccnc1)N(CCN(C(CN(CC(C)C)C)=O)C)C c1(CS(Cc2cn(-c3ccc(C)cc3)nn2)(=O)=O)ccc(C(F)(F)F)cc1C#N c1(C(=O)NCC(CC)(C)NC(=O)C2=NOC(C)C2)cnn2cccc(C)c12 N1(C(CCC2CC(C)C2)=O)CCCC1C(C)(C)CNC(=O)Cc1ncsc1Cl N1(C(CC2CCN(C(=O)NCCOC)CC2)=O)CC2COCC2(CO)C1 N1(C(C(C)SC(F)(F)F)=O)CCN(C(=O)CC23CCCN2CCC3)C(CF)C1 S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1C(C(=O)Nc2c(C)nsc2)C=CC1 C(=O)(CC(O)CC(C)(C)C)N1CCC(C(C)NC(=O)CN(C2CCCC2)C)CC1 c1(OC)cccnc1C(=O)NC(C)C(C)(C)NC(=O)CP(C)(C)=O c1(NC(C(Cc2cccs2)NC(=O)OC(C)(C)C)=O)ccncc1N1CCCC1 O(N=C1CCCCCC1)CC(=O)NC1CC(CNC(c2c(SCC)snn2)=O)C1 C1(CN(C(CSCCC(C)C)=O)C)CCN(C(C2CN(CC(C)C)C2)=O)C1 C12(NC(C3CC(NC(C=C(C)C(=O)OC)=O)C3)=O)CC1COC21CCC1 Cc1ncc(C(N2CCC23CN(C(=O)Cn2cc(Cl)c(C)n2)C3)=O)cc1C#N Cc1ccc(O)cc1CNC(C1N(C(c2ccc(Cl)cn2)=O)CCC1(C)C)=O CC(CC(=O)NC1CCC1NC(c1cncnc1)=O)C(F)F C1(C(=O)NCC2C(NC(C(CC(C)(C)C)OC)=O)CCC2)CCc2nc(C)[nH]c2C1 N1(C(COCCC=C)=O)CC(C)CN(C(c2ccoc2)=O)C(C)C1 CC1(NC(C2CC2c2ccccc2)=O)CCN(C(=O)CC2CCC2(F)F)C1 c1(C(N2CCCC(C(C)NC(c3cnc[nH]c3=N)=O)C2)=O)ccc2scnc2c1 C1(N(C)C(C2(F)CCCC2)=O)CC2CCC(C1)N2C(=O)CCCn1ccccc1=O c1(C(=O)NC2CN(C(C3CCC(=C)CC3)=O)CC(O)C2)cncc2sccc12 C1(CN(C(CC(C)OC)=O)C)CCCN(C(c2ccccc2C(C)(C)C)=O)C1 C1(C(C)(C)C)CCN(N2CCC(c3nc(=N)[nH][nH]3)C2)C1 N1(C(=O)NCCOCCCN(C)C)CC2(CC3CCCN3C=O)CCC1CC2 CCCC(CNC(=O)CCCNC(N)=O)C(=O)N1CC(N(C)C)C(C)C1 N1(C(C2C(CCC)C2)=O)C(C(=O)NCc2nc(C)sc2C)CC2CC12 C1(NC(c2c(C#N)nc[nH]2)=O)CC2CN(C(=O)C=CCN3CCCCC3)CC12 c1(CC(=O)N(C(C)CNC(c2c[nH]cc2Br)=O)CC)cc(C)ccc1F c1(C(=O)NCCCOCCCNC(C2CSC2)=O)ccncc1O CC(C)(C)CCC(=O)N1CC2CC1C2NC(C1NC(=O)OC1(C)C)=O c1(NC(C=CCC(C)(C)NC(=O)C=CC2CCCCC2)=O)cn2ccnc2cn1 C=CC(C)(C)CC(=O)NC1CCC(CC(=O)NC2C3CCC(C3)C2CO)CC1 CC1(C)CCN(C(=O)CCc2cocn2)C1CNC(c1coc(CO)c1)=O C1(C(=O)NCCCC(C)NC(c2coc3c2COC3)=O)CC(S(C)(=O)=O)C1 C(CC(C)(O)C(C)(C)CNC(=O)NCc1ccc(OC(F)(F)F)cc1C)OC C1(CC(=O)NCC2N(C(C=C(CCN(C)C)Cl)=O)CCC2)OCCC1(C)C c1(NC(C2CC23CC3)=O)cc2cc(Oc3ccccc3)ccc2cn1 CN1C(=O)CCC1C(=O)NC1(C2CCCN2C(c2[nH][nH]c(=N)c2Br)=O)CC1 c1(C(=O)NCC2CN(C(C(C)CO)=O)C3(C2)CCC3)cnc2c(C#N)cnn2c1 Cc1cn2c(C(=O)NCCCC(C)NC(=O)CC3CCCC3C)cnc2s1 C1(C)(CNC(c2cc(C)c(C)[nH]2)=O)CN(C(c2cc(O)nn2C)=O)CCO1 N1(C(CCCCCn2cc(CN(C(C)=O)C)nn2)=O)CCCC2(CC1)CC2 C1(CCNC(CC(=O)NCC)=O)COCCN1C(=O)Cc1cccc(C)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)C=CC(=O)OC(C)(C)C)CC(C)C1 N1(C(C(C)(C)N2CCCC2)=O)CCC(C2CCN(C(c3ccc(Cl)nc3)=O)C2)C1 C1(N(CCOC)C)CCN(C(=O)NC(c2ncc(-c3ccccc3)o2)C)CC1 C=C1CCNC(C(=O)NC(=O)Cc2ccccc2C)C1.c1(CC2CC2)nn[nH]n1 C#Cc1ccc(C(N2CCC(C(C)(C)C)(CNC(=O)C#CC(C)C)C2)=O)cc1F C1(C(C)O)CCN(C(c2cnc(CNC(=O)CCN3CCCC3=O)o2)=O)C1 c1(C(=O)NC(CC)CNC(=O)C(F)CSC)ccc2c(c1)NC(=O)CNC2=O C1(NC(C(CC)C(C)O)=O)CCC2CN(C(C3CC3(F)F)=O)CCC2C1 C(N=c1nc2ncn(C)c2c(NCc2cccnc2)[nH]1)c1c(C)cc(C)oc1=O CCCCC(O)C(=O)N1CCC(NC(=O)CCc2n[nH]c(=N)s2)CC1 n1(C2CCN(C(=O)Cc3ccncc3Br)CC2)nc(O)ccc1=O C1(C(=O)NC(C2(OC)CCC2)C)CC2CC2N1C(c1nnc(S)n1C)=O C1(C(=O)NC(c2cnn(C)c2)C)(C(C)C)CCCN1C(=O)CC1CCCO1 c1(C(=O)NCC2C(CC(=O)NCC3(F)CC3)C2)ccncc1O C(=O)(C#CC1CCCO1)N1CCCC(C)(NC(COCC(C)C)=O)C1 C=CCC(C(=O)NCC1CC(NC(c2cc3c(s2)CCCC3)=O)C(O)C1)C(C)C C(C1=NOC2COCC12)NC(CC(C(C)OC)NC(=O)CCn1cccn1)=O C(=O)(C(C)C(C)(C)C)NC1(C(=O)NC(c2ccn(C)n2)CC)CSC1 c1(N2CCC(CCNC(=O)CC(c3ccc(Cl)cc3)O)C2)ncnn2cccc12 c1(CN2CC(NC(c3cccc(C(N)=O)c3)=O)C(F)C2)c(Cl)ccc(F)c1F C1(CNC(c2cnc(CC)nc2O)=O)CC12CCN(C(c1sccc1Cl)=O)CC2 Cc1nc(Cl)nc(N2CC3(COC(CNC(C4CC(=O)NC(=O)N4)=O)C3)C2)c1F c1(-n2cc(C3(CCC(=O)c4ccco4)CC3)nn2)ccc(F)cc1 N1(C(C=NC(=O)CCC2CCCC2)=O)CCC2(CCC(CCOCC=CC)CC2)C1 C(=O)(CCC(C)NC(=O)C=C(CC)CC)N(CCCC=C)C C1(N(C)C(C2CC2C#N)=O)CN(C(=O)C=C2CCC2)CC1O Cc1cccc2c1N(C(c1nc(Br)c(C3CC3)s1)=O)CCN2C(C1CCCO1)=O Cc1cc(Cl)c(C(=O)NCC2CC2CNC(=O)CC2CC(F)(F)C2)cc1C c1(CC(=O)N(C2CCN(C(=O)CNC(=O)C(C)(C)C)C2)C)ccc(F)nc1 c1(NC(N(CC(=O)N(C)C)C)=O)ncc2n1CCNC2 c1(OCC)cccc(C(=O)NCC(C)CNC(C2C3C4CCC(C4)C23)=O)c1 N1(C(C2CC(C)=C(C)CC2)=O)CC(C2CCCN(C(=O)C(O)CCC(C)C)C2)C1 c1(C(=O)NCC(N(C(c2c(C)ccnc2)=O)C)C2CC2)ccc(=O)n2c1CCC2 CCCC(C)N(CCC(=O)NCCC1(NC(=O)CC2CCC2)CCC1)C1CC1 C=CC1(C(=O)N(C)Cc2cn[nH]c2)CCN(C(C2CNC(=O)C2)=O)C1 N1(C(C2CCN2Cc2ncc[nH]2)=O)CC2CCC(C1)O2 N1(C(c2ccc(C(C)=O)s2)=O)CCCCC1C1(NC(c2ccccc2Cl)=O)CC1 c1(C(N2CCN(C(=O)C=CCF)CC2CO)=O)cc(F)c(CO)c(F)c1 c1(C(N2C3CC(CC(NC(CCCC(N)=O)=O)C3)C2)=O)cc2ccc(Cl)cc2s1 N1(C(C(C=CCCC)O)=O)C(C)CC2CN(C(c3nn(C)cc3Cl)=O)CC12 c1(C(=O)NCCCN(C(CCCOC)=O)CCO)ccc(S(N)(=O)=O)c(OC)c1 c1(C(=O)NCC(CC)NC(c2c(Cl)cnn2C2CCCC2)=O)cn(C)nc1O C1(OC)CN(C(C2(C)CCCC2)=O)CC1C(=O)NCC(C)CC1CCC1 c1(C(N2CCC3C(C2)CN3C(=O)C(O)CN2CCCC2)=O)cccc2c1NCC2 c1(NC(CC2C(CNC(COCC)=O)C2)=O)cncc(Br)c1C C1(C(N(CC)CC)=O)(NC(c2c[nH]nc2C2CCOC2)=O)CC=CC1 C1(NC(CCC(=O)NCC)=O)CC2CC1N(C(=O)Cc1csc(=N)[nH]1)C2 CS(=O)(=O)C1CCCC1C(N1CC(NC(=O)Cc2cnns2)CC2(CC2)C1)=O c1(C(=O)NC2CCCC(NC(C3CC(C#N)C3)=O)C2)ccc2ccccc2c1O C1(C(=O)Nc2c(C(C)(C)C)onc2)CNCCC1(C)C c1(N(C)CCn2cccn2)nc2c(c(=NCC3CCC=CO3)[nH]1)CCCC2 CC(C)C(C(=O)N1CC(O)(CNC(=O)Cc2nnc(O)s2)C1)N1CCCC1=O N1(C(C2C(O)CCN(Cc3c(C)c(Br)ccc3)C2)=O)CCSc2ccccc21 C(c1ccccc1Cl)=CC(=O)NCC1N(C(c2cc(C(C)=O)c(C)o2)=O)CCC1 c1(C(N2CCN(C(C=C(C)Cl)=O)CC(O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N2CCC(N(C(c3c(O)cc(C)nn3)=O)C)C2)=O)cccc2c1CCC2 Cc1ncc(C=CC(=O)NC2CCC(Nc3cc(C(F)F)ncn3)CC2)s1 c1(C(N2CCC(N(C(=O)C3=NOCC3)CC#C)CC2)=O)ccc2cnoc2c1 N1(C(C(C)=CC)=O)CC2ON=C(CNC(=O)CSS(C)(=O)=O)C2C1 c1(CC(c2n(CC)c(N3CCCC(C)C3)nn2)C)ccc(F)c(F)c1 C(C(=O)N1CCCc2nccn21)=CCNC(=O)CCn1cccn1 c1(OCC)sccc1C(=O)N(CC(C)NC(=O)C(C)Cc1ccccc1)C N1(C(C(=O)NCC(c2cccc(F)c2)N(C)C)=O)CC2CS(=O)(=O)CC2(C)C1 N1(C(CN(CC(C)C)C)=O)CCC(C(=O)NOC(C)C)(C(C)C)C1.C(N)(=O)O N1(C(C=CC=CC)=O)CCC(NC(c2cn(C(F)F)c(C)n2)=O)C(O)C1 N1(CC)C(=O)CCC1CC(N1CCC(O)(CN(C(=O)CC2(C)CCOC2)C)C1)=O Cn1cc(Cl)cc1C(=O)NC(CNC(c1cccnc1O)=O)C1CCC1 N#Cc1cc(Br)ccc1C(N1CC(NC(=O)COc2ccc(Cl)nc2)C1)=O Cc1ccc(C(N2CCCCC(NC(=O)Cc3n[nH]c(=N)s3)C2)=O)c(C)c1 C1(C(=O)NCCC(C)O)CC2(CCN(C(c3ccnc4cc[nH]c34)=O)C2)C1 c1(NC(c2ccc(Br)cc2)CC)cc(C)c([N+](=O)[O-])cc1Br c1(C(=O)NC2C(CNC(=O)CCc3ccoc3)C2)cnn2c1CCC2 C(CCC(=O)NCCCN(C(=O)CCc1ccn(C)c1)C)N(C(C)=O)C CCC(C#N)C(=O)NCC1CCCCN1C(=O)Cc1cccnc1 c1(C(N2CC(C(=O)NCC3CCOC3C)(CC)C2)=O)c(C)nsc1C c1(N2CCN(C(C(n3cc(C4(O)COC4)nn3)C)=O)CC2)cncc2nnnn12 C(=O)(CCN=C(NCc1cccc(Cl)c1)NCc1cnc(C)s1)NC CCCCCCCCC(=O)N1CC(NC(=O)COCCCOC)C2(CC2)C1 c1(OC)cc(F)ccc1NC(C1C=CC(NC(c2cn(C)nn2)=O)C1)=O C12(NC(CC)=O)CN(C(=O)Cn3c(C)cc(O)cc3=O)CC1CS(=O)(=O)C2 N1(C(c2ccc(C)cc2O)=O)CCCC2(CCN(C(c3c[nH]nc3Cl)=O)C2)C1 CC1(C)C=C(C(=O)N2CC(F)(F)CC2CNC(=O)C(=Cc2c[nH]cn2)F)C1 C1(CN(C(C(CO)OC)=O)C)COCCN1C(C1CCC(N(C)C)CC1)=O C12(C(=O)NC(CCC=C)CO)CC(CN(C(c3nc(OC)c(C)s3)=O)C1)C2 N1(C(CS(N)(=O)=O)=O)CCCC2CCN(C(=O)COCC(F)F)CC12 c1(C(=O)NCC(=O)NC)ccc(NCCc2cccc(Cl)c2)nc1 C1(CNC(CCCC(C)=O)=O)C2CCCC1N(C(=O)CC1CC=CCN1C)C2 C=C(C(=O)N1CCN(C2CN(C(c3cc(C#N)ccc3Cl)=O)C2)CC1)C(F)(F)F c1(CN(C)CC2CCC(n3ccnn3)CC2)ccc(C#N)cc1 N1(C(C(CC)N(C)C)=O)CCC2(CC1)CC(NC(c1cc(Br)n[nH]1)=O)CO2 c1(C(N(C(CNC(C(C=C)c2ccccc2)=O)C)C)=O)cc(N)c(O)c(F)c1 c1(CC(C)NC(N(C(C#C)C)CCCC)=O)ccnn1C C#CCCCC(C)C(=O)NC1CC2(C1)CC2C(=O)NC1CCC12CCCC2 C12(NC(=O)Cc3cc[nH]c3)CC(C1)N(C(=O)CSCc1ccccc1O)C2 C1(NC(C(c2nc(C)sc2)=O)=O)CN(C(=O)CCN2CCCCC2)CCC1C c1(C(=O)NC(C2CCCN2C(c2nnn(C(C)(C)C)n2)=O)(C)C)ccc(Cl)o1 Cn1cnc(C(=O)NCC2(C)CCCNC2)cc1=O CC1(C)NC(=O)CC1C(=O)NCC1(O)CCCN(C(c2ccoc2)=O)C1 c1(C(N(CCN(C(C(CC)OC)=O)C(C)C)C)=O)cn2c(n1)CC(C)CC2 c1(C(N2CC(C)(C(=O)NCC3(OCC)CC3)C2)=O)ccn(C)c(=O)c1 c1(N2CC=C(C)C2)nc(N2CCC(C)(C(N)=O)C2)nc2ccccc12 c1(CC)c(OC)cccc1C(=O)NC1CCCN(C(=O)COc2ccsn2)C1 CCCC(C(O)C(=O)N1CC(N(C)CCOC)C1)NC(=O)CC(=O)OCC Cc1cc(C(=O)NCCCNC(c2ccnc(N(C)C)c2)=O)nn1C(C)C C1(C2CCCN(c3nc4cc(F)ccc4o3)C2)(NC(C2=NOC(C)C2)=O)CC1 C=CC1CCCCN1C(=O)C=C1CCOCC1.S(C(F)(F)F)CC(=O)NCC C=CC(C)(CCOC)C(=O)NCCCCC1(NC(c2ccc(C)c(OC)c2)=O)CC1 N1(C(c2scc(OC)c2)=O)CCCC2(CC(NC(c3cc(C)c[nH]3)=O)C2)C1 N1(C(CCOCCOC)=O)CCC2C(NC(C3CC(F)(F)C3)=O)CC12 c1(C(N2CC(N(C(C(C)OCCOC)=O)C)C2)=O)cccc2c1CNC2=O c1(CNC(c2ccncc2F)CC)cc(O)ccc1F C1(NC(C2CCC(C(N)=O)CC2)=O)C2CCC(C2)C1C(N1CC2CC1CS2)=O C(=O)(C(F)(F)c1csc(C)c1)NCC(c1ccccc1)COC.C1(=O)CN1 CC(O)(CNC(C1CCC(C2CC2)N1C(=O)CN1CCNC(=O)C1)=O)C(F)(F)F C1(CCNC(Cc2nc(C)oc2)=O)CCCN(C(=O)C(C)Sc2ncccn2)C1 c1(C(=O)NC(CNC(CCC#C)=O)C(C)C)ccc(F)c(Cl)n1 N1(C(CN(C(C(C)NC(=O)C2CC2)=O)CC2CC2)=O)CCc2nc[nH]c2C1 c1(NC(c2n(CC=C)nnn2)c2ccsc2Cl)sc2c(c1C=C)CCC2 C(CCC1CC1)(C(=O)NCCn1ncnn1)NC(C(C)(O)C1CCC1)=O c1(C(=O)NCC2CCCCN2C(C2CCC(F)CC2)=O)cnn2c1OCCCC2 c1(C(N2CC(NC(C=C3CCC(C)CC3)=O)C(O)C2)=O)cc(C(F)F)cc(F)c1 CCC(CC(C)C)C(=O)N1CCC(C)C1C(=O)NCc1nc(C)ccc1C c1(C(=O)NCC(COC)C)cc(Cl)cc(Br)c1Nc1ccccc1C c1(CC(CNC(NC(CC)C)=S)C)ccccc1Cl C1(C(=O)NCC2N(C(CCc3c(C)csc3N)=O)CC2)CCn2c(C)nnc2C1 C(=O)(CC(C=C)CCC)N1C(C(N2CCC(OCC#C)CC2)=O)C=CC1 c1(OC)cccc(C(=O)NC2CN(C(=O)C=C3CCC(C)CC3)CCC2F)c1F C1(C2(NC(=O)CC3(N4CCCC4)CC3)CC2)CN(C(=O)Cn2cc(Cl)cn2)CCO1 c1(OC)ccc(C(CNC(C2(F)CN(C(c3cnn(C)c3Cl)=O)C2)=O)OC)cc1 C1(NC(CCCOCCC)=O)C2CC3C1C3C2C(N1CCC(O)(C(C)C)C1)=O c1(C(=O)NCCNC(=O)Cc2ccc(-n3cnnc3)cc2)cnn2c1OCC2 C(CN=c1[nH]c(=NC(C)CCn2ccnc2)[nH]c2c1CC(C)CC2)N(CC)CC C1(C(N2C(CNC(CCC(C)OCC)=O)CCC2)=O)C2CCCCCCC12 C(=O)(CC(C)(O)C(F)(F)F)N(C1CCN(C(c2cncc(O)c2)=O)C1)C N1(C(c2c(N)nccc2)=O)C2CCC1CC(CCNC(C1CCCCS1)=O)C2 C(C(CC(=O)N1CC2C(Cc3cccs3)C2C1)CC(C)C)NC(C)=O n1(CC(CC)O)cc(C2CC(NC(C3CSCCS3)=O)C2)nn1 C(C1CCCCC1)=C(C(=O)N(CC(C)N(C(CC(C)C)=O)C)C)F C1(c2n(CC(=C)C)nnn2)(NCCCC2CCOCC2)CCS(=O)(=O)CC1 C1(CC)CCCC(N(C(C2CC(F)(F)CN2C(=O)CCC(=O)C2CC2)=O)CC)CC1 CCCCC(C(=O)N(C(C)CNC(=O)CC1(O)CCC1)C)ON=C(C)C C(=O)(CC(F)(F)F)NC(C)C(N1CC(F)(CNC(C2CCCCO2)=O)C1)=O c1(C(=O)NC2C(CNC(C(C(C)(C)C)N(C)C)=O)C2)csc(=NC2CC2)[nH]1 CC(CNC(=O)Cc1cncnc1O)C(F)C(=O)NCCCC(N)=O C1(CNC(C2CC2(Cl)Cl)=O)CCCCN1C(=O)CC12COCC(C1)C2 N1(C(c2c[nH]c(=NC)o2)=O)CC2CC(C1)C2NC(=O)CC(C)c1ccncc1 Cc1cnc2nccc(C(N3CC4CC4(CNC(C4CC4(Cl)Cl)=O)C3)=O)c2c1 C1(C(N2C(CNC(C=CC(=O)NC3CC3)=O)CC2)=O)CCCCC1 CC1(C)CCOC(C(=O)NCCCOCCNC(=O)CSc2cccs2)C1 N1(C(c2c(SC)cccc2)=O)CCN(C(C2(C3(O)CCC3)CC2)=O)CC(C)C1 C(C)(C)(CCC(=O)NC1CCCC(NC(c2ccc(C#N)[nH]2)=O)C1)N(C)C n1(CCOCC)cc(C2CCN2C(=O)C(C)OCOC)nn1 N1(CC(=O)NC(c2cccc(C)c2)CC)CCOC2CNCC12 C1(CNC(C2C(CC)CCO2)=O)CCCC12CCN(C(=O)C=C1CCC1)CC2 N1(C(CC(CCC)(C)O)=O)CCN(C(C2CCC(=O)N2)=O)CC12CCC2 C(CC(C(=O)N(C(CC)C1CC1)C)NC(=O)CC1CC(C)(C)CO1)=CC c1(CCCCCC)nc(CCOCCOC)n(-c2ccc(F)cc2)n1 C1(CC(=O)NCCCN(C)C(c2ccc(CO)s2)=O)CCCS1(=O)=O C1(C(=O)OCC)OCCNCC1NCC.C(CO)(C(C)C)S(=O)(=O)Cc1cnc(Br)o1 c1(N2CC3C(CNC(CCCC#C)=O)C3C2)ncc2c(ccn2C)n1 CC1(NC(=O)Cc2cnsc2)CCN(C(=O)Cc2nc(-c3cccs3)no2)C1 c1(CC(=O)NCC(CC)NC(=O)C(C)=CCO)cn(C)nc1C(F)(F)F c1(CCC)n[nH]cc1C(=O)NCC(C(C)C)NC(c1c[nH]nc1C(C)(C)C)=O N1(c2cc(C)nc(N3CCC(n4nccc4C4CC4)C3)n2)CCC(N)C(C)(C)C1 O=C(CCCC1CCC1)NC(c1ccoc1)CNC(c1ccco1)=O N(C(=NCC1CCCO1)NCC(c1ccsc1)O)Cc1ccc(C(=O)OC)o1 c12cccc(c1)N(C)C(=O)CN2.c1(C2(CN(C)C)CC2)ccccn1 C1(C)(NC(C(n2cc(Cl)cn2)C)=O)CCCN(C(=O)C(N2CCC(C)CC2)=O)C1 N1(C(C2C(C#C)C2)=O)CCC2(CC1)CCN(C(C1CCc3ccnn3C1)=O)CC2 CC1(C)CC(NC(C2CCCCS2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)C1 CC(C)C(C(=O)NC1CN(C(C2(OC(N)=O)CC2)=O)CC1C(F)F)NS(C)(=O)=O Cc1ncc(-c2cncc(C(N3CCOCC3)=O)n2)cn1 CC1CN(C(=O)C=C2CCN(C)C2)CC1CN.c1(CC(=O)N(C)C)ccccc1 C1(CNC(=O)Cn2nnc(=O)[nH]2)CCCCN1C(C1CCCC12CC2)=O c1(C(N2CCCC(N(C(COCCOC)=O)C)C2)=O)cc2ccc(Cl)nc2s1 Cc1ccn2c(=O)c(C(=O)NC3CCCCC3NC(C3CC(O)C3)=O)cnc2c1 CCC(O)C(C)C(=O)NC1(C(=O)NC(C)CC(C)(C)C)CCCCC1 c1(C(N2C(C(N(CC)CC3CCCO3)=O)C=CCC2)=O)ccccc1C#N C(=O)(CC(C)C)N(C(CCNC(C1CC(C(=O)OCC)C1)=O)C)C CCC(CC1CC1)C(=O)N1CCC(N(C(=O)CC#N)CC2CC2)CC1 C(=O)(CCCCC(=O)N1CC2CC1(C(=O)NC1CC1C1CC1C)C2)OC c1(C(=O)NCC(C)N(C(C2CCCCC2O)=O)CC)ncc(C)cc1OC c1(C(=O)NC(C(=O)N(C2CC3(CC3)C2)C)CO)ccnc(C(=O)N(C)C)c1 C1(N(C(CN(C)CCN(C)C(c2ncccn2)=O)=O)C)CCCC(C)(C)C1 N(C(=NCc1ccccc1CO)NCc1cc(C)n(C)n1)C(C=C)C Cn1ccc2cccc(C(N3CCC(N4CCCCC4)C3)=O)c12 C1(C(=O)Nc2cn(C)nc2-c2cccc(F)c2)C2Cc3cc(Cl)ccc3C12 C1(NC(C2C(C(C)NC(C(C)(CO)OC)=O)C2)=O)Cc2cscc2C1 C1(CNC(c2c(C)cns2)=O)CN(C(=O)Cc2csc(C(C)(C)C)n2)CCO1 C1(C(=O)NC2C(NC(c3ncc(C)cc3C)=O)CCCC2)CCc2c[nH]nc2C1 CCC(C)CC(=O)C(=O)N1CCC(C(=O)N(c2cccc(F)c2)C)C(C)(C)C1 c1(OC)cc(F)c(NC(=O)CC2CN(C(c3cc(C)cc(F)c3N)=O)C2)c(Cl)c1 c1(NCc2n(C)c(Br)nc2)ncccc1S(=O)(=O)Nc1cccn(C)c1=O c1(CNc2n(C)ncc2[N+](=O)[O-])cnc2c(c1)ncn2C.C12CC(C1)CNC2=O N1(C(=O)Nc2c(CC)cccc2)C2CCC1CN(C(C1CCCS1)=O)C2 N1(C(C2C(c3c(C#N)cccc3)C2)=O)CCC2CCC(C1)N2C(=O)C(N)=O CCCCC(O)CC(=O)N1CCC(C)N(C(c2nc(C)sc2Br)=O)CC1 CCCCC(C(=O)NCc1cc(C(N)=O)co1)NC(c1nccs1)=O C#Cc1cnc(C(=O)NC(CCNC(=O)C(C2CCCCC2)O)C(C)C)c(C)c1 N(C)(C(=NCCC#N)NCC1CCN(C(=O)OC(C)(C)C)C1)C(CCC)CO c1(C(=O)OC)cnc(CNC2(c3cccc(Br)c3)CC2)nc1 C(=O)(CCCCCC(C)O)NCC(C)(C)NC(COCCC#C)=O CC1(C)CCC(N=c2[nH]c(=NCCC34CCCC3C4)c3cc(F)cc(F)c3[nH]2)C1 c1(C(=O)NCC2(CNC(C34CCC(CO3)C4)=O)CCCC2)ccn2nnnc2c1 C1(C(N(CCC(=O)NCC2(CCO)CC2)C)=O)OCCC1(C)C C=CC(C)(C)C(=O)NCC1CCCN(C(=O)CC23CCCC2C3)C1 Cc1c(O)ccc(C(=O)NC2CCCC(NC(=O)C(O)C3CCCC3)C2)c1C C(C(CNC(c1cc2occc2s1)=O)C(F)(F)F)NC(c1nc(C)nn1C)=O c1(SC)nc(N2CCC(C(=O)Nc3cc(C)no3)C(O)C2)ncc1Br C1(O)(CC(=O)NCc2ccc(C(=O)NCCN(C)CCO)s2)CCOCC1 C1(C(=O)NCCCOCCNC(C2(CF)CC2)=O)CC2CCC(C1)S2(=O)=O N1(C(C(COC)COC)=O)C2CCC1(CNC(C1CCCC1C(=O)OC)=O)CC2 N1(C(COC)=O)CC(N=c2[nH]c3c(c(=NCCCn4nccn4)[nH]2)COCC3)C1 c1(C(=O)NCCCCNC(c2ncncc2Cl)=O)c(C(F)F)cccc1Cl c1(C(=O)NCC2C(NC(=O)CC3(O)CCCCC3)CCC2)ccn2nncc2c1 C1(NC(C(CC=C)CC)=O)CCC2(CC1)CN(C(C1(CCCF)CC1)=O)CCO2 c1(C(=O)NC)cccc(C(N2CC(OC)C(F)C2)C(=O)NCCCSC)c1 N1(C(C2N(CC)CC2)=O)CCCC1CNC(=O)CCc1cn(C)nn1 c1(OC)cc(Cl)c(Cl)cc1C(N1CCCCC1CCCNC(=O)CC(C)(C)O)=O c1(CC(=O)NC2C(CNC(CCc3cc(C)[nH]n3)=O)C2)ccc2c(c1)OCO2 C1(NC(Cc2n(C)cnc2)=O)CC2CN(C(=O)C3=CS(=O)CCC3)CC2C1 N1(C(C(C)C(C)(F)F)=O)CC(CNC(C2CC(N=[N+]=[N-])C2)=O)CC12CCOCC2 C(=O)(C(CNC(C1CC1Cl)=O)C(C)(C)C)N(CCC)C N1(C(c2n(CC)ccn2)=O)CCN(C(=O)CC(C)COC)C(CF)C1 c1(C(N(C(CCNC(C=CC(=O)OCC)=O)C)C)=O)nnn(C)c1CC c1(C(=O)NC2CC(C)(NC(=O)C=CCF)C2)ccnc(CO)c1 C1(C(=O)Nc2c(C(=O)OC)c(C)on2)Cc2cc(Br)ccc2O1 CC(C)(C)CCC(=O)N1CCC2C(NC(=O)Cc3cccc(NS(C)(=O)=O)c3)C12 Cc1nonc1CNC(=O)C(CO)NC(=O)C(C)c1ccco1 C1(NC(C(C=C)C)=O)CN(C(=O)C(C)n2ccnn2)CC1F CC(C)C(C)(CNC(=O)CSc1ccoc1)NC(=O)COC1CCCC1 C1(C)(C(NOCC2CC(=C)C2)=O)CCCN(C(c2ncccc2F)=O)C1 Cc1ccn2c(C(N3CCC(NC(=O)CCC4CCC(=O)N4)C3C)=O)cnc2c1 c1(C(N2CC(NC(c3cc(F)c[nH]3)=O)C3C2C3)=O)cccc2ccccc12 Cn1c(C2CCCN(C(C3OCCC4CNCCC34)=O)C2)nc2ccccc12 c1(C(N(C2CN(C(C3CCN(C4CC4)CC3)=O)C2)C)=O)ccnnc1O C(N=c1nc2c(cnn2C)c(NC2CCOC(C(C)(C)C)C2)[nH]1)c1c(C)c[nH]n1 C1(C)(C(N2CCC(CC(=O)N(C(C(C)SC)C)CCC)C2)=O)CCCN(C)C1 Cc1cc(F)c(C(N2CCC(F)(C(=O)Nc3cnccc3C(N)=O)C2)=O)cc1Br c1(C(=O)NC(CNC(CC2C(C)(C)C2)=O)CO)cccc(C2CC2)c1Cl C1(CC=C)(C(N2CCC(N(C)CC)C2)=O)CCCC1.N12CC(C1)C2=O C1(C(=O)NCCN(C(C(C)=C2CC2)=O)CCCN(C)C)NC(=O)CC1C c1(C(C(=O)NC(C)CCNC(=O)C(O)C2CCCC2)C)ccc(Br)cc1 C=C1CCC(C(=O)NCC(C)(CNC(=O)C(C(C)C)N(C)C)OC)CC1 Cc1cc(C(=O)NCC2(CF)CCC2)c(O)nn1.N12CCCC(C1)C2=O CC(C)(C(=O)NC1CC(C)(NC(C2CC3OC2C2CC32)=O)C1)S(=O)(=O)C1CC1 N1(C(CCC)=O)CC2(CCNC(=O)CC(C)c3cnn(C)c3)CCC1C2 c1(C(N2CCCN(C(=O)CSC3CCS(=O)(=O)C3)CC2)=O)cn2c(n1)CCC2 N1(C(c2c(C)c(C(F)(F)F)ccc2)=O)CC2CCC(C1)N2C(=O)C(C)(C)Br N1(C(=O)CC2CCN(Cc3ccccn3)C2)CC2CCCC2C1 c1(C(N(C2CN(C(C3CCCC3(C)C)=O)CC2O)C)=O)ccc2ccncc2n1 C1(NC(=O)C=Cc2cccs2)CCCC12CN(C(c1occc1F)=O)C2 CON1CCC(NC(C2CC3(CC3)CN2C(C2CCC(C3CC3)C2)=O)=O)CC1 C#Cc1ccc(C(N2CCC(C(=O)N(C(CC)C3CC3)C)C2C)=O)cc1C C(C(CC(F)(F)F)NC(=O)C(C1CC1)C1CC1)NC(C(C1CCC1)OC)=O c1(N(C(c2cncnc2)C(=O)NCCCOCCO)C)c(Br)c(Cl)nn1C N1(C(CC2ON=C(C)C2)=O)CCCN(C(c2cnc3n2CCCC3)=O)CC1C N1(C(C2CCN(CC)C2)=O)CCC2(C1)CN(C(c1cc(C(N)=O)n[nH]1)=O)C2 c1(CC(N2C(CC)CN(C(=O)CC3CC3(C)C)CC2)=O)ccc2ccccc2c1 N1(C(C2CCN(CC)C2)=O)CCC(C(=O)NC(C2CSC2)C)CC1C c1(C(=O)NC(CN(C(=O)C(C)(O)c2ccccc2)CC)C)nnn(CC)c1C C(=O)(CCCN=[N+]=[N-])N1CCCC(CN(C)C(c2cnc(O)n2C)=O)C1 c1(C(=O)NC2C(C)CCN(C(C(C)OC)=O)C2)cc2c(s1)COCC2 N1(C(c2c(C)[nH]c(C)c2C)=O)CCC(C)(C)C(NC(c2ncccc2F)=O)C1 c1(C(=O)NCC(CNC(C(C2CCC2)OC)=O)OC)cccc2nn(C)cc12 C1(CCC)CCCC1C(=O)N(CCN(C)C(c1cnoc1C(C)C)=O)C(C)C CC1CCC(C(=O)NCCC(O)CNC(=O)Cc2sccc2Br)CC1 C1(c2cccc(C)c2)CCN(C(=NCCC(C)C)NCC23CC=CC(C2)OC3)C1 c1(C(=O)NCC23N(C(C(C)OCCOCC)=O)CC(C2)C3)cc2sccc2[nH]1 C(=O)(CC(C)(C)CNC(=O)Cc1cc(CO)on1)NC(c1ccco1)CC S1(=O)(=O)c2ccc(c(Cl)c2)CN1Cc1cccc(C(C)C)c1.C(COC)OC c1(CCC(=O)N(CC(C)NC(=O)Cc2scnc2C)CC)c(C)nc(C)nc1O C=C(C)CC(C(=O)NC1CC1CNC(=O)Cc1ccnn1C(C)C)OC n1(CC(=O)NCC(C(C)C)NC(=O)CC(C)n2cccn2)ccc(=O)n(C)c1=O C12(C(=O)NCC(C)F)CCC(NC(C3CNC(=O)CC3C)=O)(CC1)C2 c1(C(N2C(CN(C(C=C(COC)C)=O)C3CC3)CCC2)=O)ccc(OC)nc1 c1(C(=O)Nc2c(C)nn(CC)c2C)c(OC)cc(OC)cc1N C1(NC(CC(CC)CN(C)C)=O)CC2CC1CN(C(c1cc(C)ncc1Cl)=O)C2 C1(NC(CCCC=C)=O)CC2CCC1N2C(c1cnn(C(C)C)n1)=O C(=O)(C(C)(COC)CC)NC1CCN(C(c2cn(CCC=C)nn2)=O)CC1 c1(OC(C(=O)N(C2CCN(C(=O)CCF)C2)CC)C)ccc(C)cc1C C(=O)(C1=NOC(C)(C)C1)NC1(CC=C)CCN(C(C2(F)CCC2)=O)C1 C#CCCCC(C)C(=O)N1CC(F)(CNC(c2cn3ccsc3n2)=O)C1 C1(C(=O)OC)(OCCNC(=O)CC2CCC(C3CC3)O2)CCC(C)C1 C(N=c1nc[nH]cc1C#N)C1C(NC(CSC)=O)C2(CC1)CCC2 N1(C(C=C(C)C2CC2)=O)CCCC2C(NC(C3COCC(C)O3)=O)C(C)(C)C12 C=CCCC(C)C(C(=O)NCc1nnn(C)n1)N1CCC(c2ncccn2)CC1 N1(C(C=C(CCC)C)=O)CC(C(=O)N(CC(C)O)CCF)CC(C)C1 C(=O)(CC(C)(C)c1cccs1)NCC(CCOC)NC(c1ncn(C)c1C)=O N1(C(CNC(CC)=O)=O)CC2CC(C1)C2NC(c1ncn(CC)n1)=O Oc1cc(C(c2nnnn2Cc2ccccc2)NC2(CCO)COC2)cnc1Br C=Cn1nccc1C(=O)NC(CNC(C1(c2cccnc2)CC1)=O)CC N1(C(C(C)=C2CCC2)=O)CCC(C(=O)NCCCC2(O)CCC2)CC1 n1(C(C)C)ncc(C(=O)NCCC2(NC(=O)CC3CCOC3C)CCC2)n1 CC#CCC(C(=O)NCCOC1CCOC1)NC(c1c(CO)n[nH]c1C)=O C(=O)(C(C)(C)F)N(CCCN(C)C(C1CC1(C)C(F)(F)F)=O)C CCCCC(CC)CC(=O)N1C2CCC1C(CNC(=O)Cc1ccccc1F)C2 Cc1nc2sc(C(=O)Nc3ccc4nnc(C(F)F)n4c3)cn2c1Br C1(C(=O)NCC2C(C)CN(C(=O)C=CCF)C2)CC2(C1)CC(O)C2 CC(C(=O)NCCCC1(NC(C2SCCS2)=O)CC1)C(C)c1ccc(F)cc1 C(=O)(C(F)(F)C(F)(F)F)N(C1CC(NC(=O)Cn2ccc([N+](=O)[O-])n2)C1)CCO C1(C(=O)NCc2occ(C(N3C(CC)CC3)=O)c2)CCCCC1F N1(COC)CC(C(=O)NCC(C)NC(c2cc(F)ccc2Cl)=O)CCC1=O c1(N(CCO)C2CC2)cn(C2CCOCC2)nn1 C(CCCC(=O)NCC1CCCN1C(=O)Cc1n[nH]c(=N)s1)SC Cc1cc(CCC(=O)NCC2COC(CNC(c3n[nH]cc3C)=O)C2)on1 c1(OCC)cc(N(CCCN(C(=O)CN2CC(=O)N(C)C2=O)C)C)nc(C)n1 Cc1cc(C)cc(S(=O)(=O)N2CCOCC2C(=O)Nc2ncnc(C)c2C#N)c1 C1(NCC2(C(=O)NCC3(C(C)C)CCCCC3)CCCO2)CCCCC1(C)C Cc1ccc2[nH]c(CN3CCC(C(=O)Nc4nc(O)cs4)CC3)cc2c1 N1(C(CCCC(CC)NC(=O)C(C)(C)CC2CC2)=O)CCCCCCCCC1 c1(C(N2CC(OCCNC(C3CC(CC)C3)=O)C2)=O)cc2ccccc2nn1 O=CN1CCCC1C(N1CCC(O)(Cn2cc(-c3cccs3)nn2)C1)=O N1(C(C(COC)OC)=O)CCC(C2(O)CCN(C(=O)CCNC(=O)CO)C2)CC1 N1(Cc2ccc(S(CC)(=O)=O)s2)CCC2C(=O)NC(=O)C2C1 C1(N(C(c2scc(OC)c2)=O)C)CCN(C(C2(O)CC(C)(C)C2)=O)CC1C C(CCC(C)C(=O)N1CCC(N(C)C(c2cc(OC)ns2)=O)CC1)OC N1(C(C(CC)(C)C(F)F)=O)CC2(C1)CN(Cc1c[nH]ccc1=O)CCO2 C1(CN(C(Cc2cnc(C)o2)=O)C)CCCN(C(C2(C(C)C)CCC2)=O)C1 c1(N2CCCC(C(=O)NCC(C3CCCO3)O)C2)ncnc2ccccc12 Cc1oc(CO)cc1C(=O)NC1CCCC(CNC(C2(Cl)CC2)=O)C1 C1(CNC(C(=O)NCCC(C)(C)CNCc2ccccc2)=O)Cc2nccn2C1 CC(C)CC(O)C(=O)NCc1ccccc1CN(C(=O)CCc1cnn(C)n1)C C1(CC)CN(C(c2cc(CNC(=O)CC(C)OC)ccn2)=O)CCS1 N1(C(C(=O)NCC#C)OCC2(SC3CCC3)CC2)CCN(C)C(CC(C)C)C1.COC C(=O)(C(CNC(=O)CCC1CC1(F)F)CC1CC1)NC(CC)C(=O)NC n1(C(C)(C)C)ncc2c(N3CC4C(Nc5ncnc(O)c5Br)C4C3)ncnc12 c1(C(N2C(CN(C)C(c3cnn4c3CCC4)=O)CCC2)=O)cc(=O)cc(Cl)[nH]1 C1(C)(NC(C2(COC)CN(C(=O)C(F)C3CCOC3)C2)=O)CN2CCC1CC2 c1(OC)cc(OC)nc(N2CCOCC(CNC(=O)Cc3cncn3C)C2)n1 c1(C(=O)NC2N(C(c3cc(OC)nc(Cl)c3)=O)CC2)ccc2c(c1)N(C)C(=O)C2 N1(C(C(C=C)CC)=O)CC2CC(NC(=O)CC(C)(C)O)CC(C2)C1 C1(C(=O)NCC(c2ccccc2)NC(c2occc2C)=O)(CC)CC1(F)F C1(NC(C(N(C)C)C2CC2)=O)CCCN(c2nnc(C(F)F)o2)C1 c1(CCC(=O)NCCOCCNC(C2OCC(C)C2)=O)ccc(F)nc1 c1(NC(CCN(C(c2ccc(CC)[nH]2)=O)C)C(C)C)ncnc(Cl)c1[N+](=O)[O-] C(c1ccc(Cl)cc1F)=CC(=O)NCCOCCN(C(CNC(C)=O)=O)C C(=O)(C(F)(F)CO)NCCC1(CNC(Cn2cc(C(C)=O)nc2)=O)CC1 C(C(C(C)C(C)C)NC(=O)CN(C)CCO)NC(c1c(CC)n(C)nc1)=O C1(C(=O)NCc2ncccn2)(NC(CCCNC(N)=O)=O)CC(F)(F)C1 N1(C(CC(C(=C)C)OCC)=O)CCC(C)(C)C(C(=O)N(C)OC)C1 CCCC(CCC)CC(=O)NC(C(=O)NCC(CC)(CC)CC)C1CCC1 c1(C(=O)NCC(CNC(=O)C(C)(C)c2ccncc2)OC)nnc(S)n1C Cc1cc2n[nH]cc2cc1-c1cnn2ccc(C(=O)NCC(C)(C)CO)cc12 c1(CCC)ccc(C(=O)NC2CC(C)(C(N3CCC(C)(O)C3)=O)C2)cc1 c1(CNC(C(C)OCC(C)C)=O)ccc(C(=O)NC2C3CCCC23)cn1 CC1CCC(C(=O)NCC23CCCC2CCC3)CN1C(=O)C(F)C(F)(F)F C1(CCNC(C2CCC2CF)=O)CCCN1C(c1cnn(CC(F)(F)F)n1)=O N1(C(C(C)(C)CC#N)=O)CCC2CC(NC(c3cccc(F)c3F)=O)CCC2C1 c1(C(=O)NC2CC(C)N(C(C3CC(C(F)(F)F)C3)=O)CC2)nc2cccnc2s1 N1(C(C(C2CCC2)OCC)=O)CCC2CN(C(c3cn(C)cc3C)=O)CC2C1 c1(C(=O)NCCC(C)NC(c2cc(=N)[nH]c(Cl)n2)=O)cc(S(N)(=O)=O)c[nH]1 C1(CNC(CC2ON=C(C)C2)=O)CCCCCN1C(c1occc1C)=O N1(CC(=O)NCCNC2(C(=O)NCC3(C)CC3)CC2)CCCC1=O n1(CC)cc(C(=O)N(CCN(C(=O)CCC2(C)CC2)C)C(C)C)cn1 CC1(NC(C2CSCCS2)=O)CCCN(C(c2ccnc(OCC3CC3)c2)=O)C1 c1(C(=O)NC(CCCC)CNC(c2csc(C(N)=O)n2)=O)sc2nccn2c1C C(=O)(CCS(C)(=O)=O)NC(C1N(C(c2ccc(OC)cc2)=O)CCCC1)C N1(C(C2(CNC(=O)Cc3ccnc(Cl)c3)CCCO2)=O)CC2(CNC(=O)OC2)C1 C(C(=O)N(C)OCC(F)(F)F)N(C1CCN(C(C2(CCCC)CCC2)=O)C1)C N1(C(CC(CC2CC2)NC(CCCC(=O)OC)=O)=O)CCc2c(C)cccc21 c1(C(=O)NCC(CN(C)C(c2cnn(C)n2)=O)O)cc(F)ccc1Br c1(C(=O)NC2CN(C(c3ncc(NC)nc3)=O)CC2O)cc2c(Cl)cccc2[nH]1 N1(C(COCC(=C)C)=O)CC(C)CN(C(c2cc3ccccc3s2)=O)C(C)C1 N1(C(C(=O)NC2(CC=C)CN(C(=O)C(C)C3CCC3)C2)C)CCC(O)CC1 C(N=c1[nH]c(=NCCCC(F)(F)F)[nH]c2cc[nH]c12)c1ccc(N)c(CO)c1 Cc1nc(O)[nH]c1C(=O)N(C)CCOCCNC(c1csc(-c2cn[nH]c2)c1)=O C(=O)(CC(F)(F)C(F)(F)F)NC1CC2(CN(C(CCC(=O)NC)=O)C2)OC1 N1(C(c2nnc(C)s2)=O)CC(NC(c2cnc3ccoc3c2)=O)C(N=[N+]=[N-])C1 C1(CC#C)CN(C(=O)CCCNC(=O)CN2CCN(C)CC2)CCO1 n1(CC(=O)NCCN2CCN(C3CCN(CC)C3=O)CC2)ccc2ccccc12 C1(C(=O)NCC=C)CN(C(=O)C(C)CSC)CCO1 C(CC(C)(C)C(=O)NCC1(CCO)CN(C)C1)NC(c1ncc(NC)nc1)=O C1(C(N2CC(O)(C(CNC(C(C)N3CCC3)=O)(C)C)C2)=O)CC2C=CC1O2 CC1(C)CC(C(=O)NOCC(=O)NCC2(c3ncc[nH]3)CC2)(CO)C1 C1(C(=O)NC2C(C(C)C)N(C(c3cc(Cl)cc(Cl)c3)=O)CC2)CC2C(C1)C2(F)F N1(C(c2ccc(C#N)nc2O)=O)CCCC12CCN(C(=O)CC(F)(F)F)C2 C1(CNC(CC(=O)N(C)C)=O)COC(C)(C)CN1C(C1CC(C2CC2)=NO1)=O c1(CNC(CCNC(=O)NC)=O)ccoc1C(=O)NCC1CC1C(C)O c1(C(=O)NCC(CN(C(C2C(OC)CCC2)=O)C)C)ccc2cnccc2c1 Cc1nnc(O)c(C(=O)NC2COCC2CNC(=O)CSCCC(C)C)c1C c1(OC)ccc([N+](=O)[O-])c(CN2CCC(O)C(C(=O)NCC(C)(O)CO)C2)c1 C(=O)(CC1c2ccccc2C=CN1C(c1ccc(I)c2c1OCCO2)=O)OC N1(C(c2c(C(=O)OC)cn(C)n2)=O)CCN(C(c2cn(C(C)C)nn2)=O)CC1C C1(NC(C2CCC(=C)CC2)=O)CC=C(C(=O)N2CC(C)(C)CC2CO)C1 C1(C(C)C)CN(C(=O)CN(C2CCCCC2)C)CCN1C(c1ccccc1)=O C1(NC(C=CC(C=C(C)C)=O)=O)CCCC(NC(=O)C=CC2CCCCC2)C1 C1(C(N2CC3C(CNC(Cn4ncc(CC)c4)=O)C3C2)=O)CNC(=O)CC1(C)C N1(C(c2ccc(CCCCC)o2)=O)CCCC(C)(CNC(c2ccnn2C)=O)C1 CCCC(C)C(C)Nc1cc(NC2CCCC2CCO)ncn1 C(=O)(CCCCCCCCCO)N1CC(CN(C(CC)=O)C)OCC1 C(CC(F)F)(C(=O)NCCC1NC(=O)NC1=O)N(C)C(c1cc(C2CC2)on1)=O C1(F)(CNC(C2CCCC2)=O)CCN(S(=O)(=O)Cc2ccccc2I)C1 c1(OC)cc(F)ccc1-c1cccc(OC(c2ccc(O)cn2)=O)n1 C1(C(=O)Nc2c(C#N)nc(C)o2)CC2CCC1N(Cc1cccc(C3CC3)c1)C2 S(=O)(=O)(c1ccc(C(N2CC(N(C(=O)CNS(N)(=O)=O)C)C2)=O)cc1)NCC=C Clc1ccccc1Cc1n(-c2ccc(NC3CCOC3CC3CC3)cc2)nnn1 N1(C(c2[nH]cc(C)c2)=O)CCOCC1CC(=O)NOCCc1ccccc1 C1(NC(c2cn(C)nc2)=O)CCN(C(C2CCC2c2ccc(F)cc2)=O)CC1 N1(C(CN(C)C)=O)CCCC(CNC(c2ncsc2-c2ccccc2)=O)C1 CCCC(C#N)C(=O)N1CCC(CNC(c2ccon2)=O)CC1C Cc1noc(N)c1C(N1CC(C)(NC(=O)COC2CCCCC2)C1)=O N1(C(CCCCC(=O)OC)=O)CCN(C(=O)CC2(OC)CC2)C2COCC12 C(=O)(C1=CCN(C(=O)C=CC2CCCC2)CC1)N(CC(C)(C)C)CCC C(CC(C)C)(C(=O)NCC1(C)CCN(C(=O)CNS(N)(=O)=O)C1)OC C1(NC(c2n(CC)nnc2)=O)CN(C(=O)COCc2ccnn2C)CC1C1CC1 C1(c2cccc(Cl)c2)(Cn2cc(CCC(CC)O)nn2)CCOCC1 C1(NC(C=CCCC)=O)CCCN(C(=O)C(C2(OC)CCCCC2)(F)F)CCC1 C1(C(=O)NCC(C)(C2CC2)NC(C#CC(C)C)=O)CCCCN(C)C1=O c1(OC)ccc(S(=O)(=O)N2CCN(C(c3c(Br)ccc(C)c3F)=O)CC2C)cn1 C1(C(N(CC(F)F)C)=O)CC12CCN(C(c1cncc(OC(C)(C)C)c1)=O)C2 c1(COC)nc(C)c(C(N2CC(O)CC2C(N2CC(C)(O)C2)=O)=O)s1 C1(NC(CC2CN(C(c3c(C)noc3C)CC)C2)=O)CCCCC1C1CCCO1 N1(C(c2c[nH]c(=NC)s2)=O)CCC(C)CC1CNC(c1cnn(C(C)(C)C)c1)=O C1(C(=O)OC)CCN(Cc2cn(CC(C)N(C)C(c3ccsc3C)=O)nn2)CC1 C=C(CN=c1ccnc(NCC2(N(C)C)CCSC2)[nH]1)C1CCOCC1 N1(C(c2n(C)nc(O)c2)=O)CC(CNC(C2CC(=O)N2)=O)C(C)(C)C1 Cc1cccc(CS(=O)(=O)NC(=O)CN2CCOCC2)c1.c12ccccc1OC2 CCC(C)(CNC(=O)COc1ccsn1)C(=O)NCc1ccc(CN(C)C)cc1 C1(CC(=O)NC2(N(C(=O)Cn3ccnn3)C)CC2)CCCC2CC12 N1(C(CCNC(=O)CCCCF)=O)CCc2ccccc2C1C(=O)OC(N)=O c1(OC)ncc(C(=O)NC2CCCC2NC(=O)C(C)NC(c2ccco2)=O)nc1C C(CCN(C(=O)CSc1nc[nH]n1)C)(C(C)(C)C)NC(CC(CC)OC)=O C12(C(=O)NC34CC(NC(Cc5cc(CC)no5)=O)(C3)C4)OCCCC1C2(F)F CC1CCC(=CC(=O)NC2CCC(C)(CNC(=O)CCNC(=O)CO)C2)CC1 C(=O)(CC=C(Cl)Cl)NC(C(=O)NCc1c(CC)nn[nH]1)Cc1ccco1 N1(C(c2cc(=O)cc[nH]2)=O)CCCC2(C1)CN(C(C1CC3(CSC3)C1)=O)CCO2 C1(C(=O)NCC2N(C(c3ccc(SC)o3)=O)CCCC2)CCCC12OCCO2 N1(C(c2cccc(CC)n2)=O)CC(C(N2CCOCC2CC(N)=O)=O)C(F)(F)C1 CCCC(CC)CCC(=O)NC1CC(NC(=O)C(C)SC(C)(C)C)C1 C1(C(N2CCC(OCCNC(C=CCOC)=O)C2)=O)C(Cl)(Cl)C12CC2 N1(C(CCc2c(C)nn(C)c2)=O)CCC(NC(=O)CC2C=CS(=O)(=O)C2)C1(C)C c1(CCCOC(c2onc(C3C(N)CCC3)n2)=O)ccccc1OCC(F)(F)F C1(CCC(=O)NCCCN(C(CC2CN(C(C)=O)C2)=O)CCO)CCCC(=O)N1 c1ccccc1S(=O)(=O)C(F)(F)F.CC1(C)C=CC(C(=O)N)CC1 CC#CCCC(=O)NCC1(C)CCN(C(c2cn(-c3c(C)n[nH]c3C)nn2)=O)C1 N1(C(c2[nH]cc(CC)c2)=O)CCC2CN(C(c3cccc4nonc34)=O)CC2C1 CC1(CNC(=O)Nc2ncc(F)cc2I)CCCC(=O)N1 c1(C(N2C(CNC(C3C(C)=CCS3)=O)CCC2)=O)noc(C)c1C#N C(CCCCCCCCCCO)NC(CC1CCCN(CC=C)C1)=O c1(C(N2C(C)CCN(C(C(CC=C)C)=O)CC2)=O)cc(OC)cc2c1OCC2 C1(CNC(N(C)CCOCCN(C)C(C2(F)CCC2)=O)=O)CC2(CCCO2)C1 N1(C(C(Br)=C(C)C)=O)CCOC2(CCN(c3ncc4c(ncn4C)n3)CC2)C1 N1(C(COCCOCCOC)=O)CCCC(NC(C2(C)OCCO2)=O)C1 C=CC1CN(C(C2OCCC2CNC(C2C(C#N)C2(C)C)=O)=O)CCO1 c1(C(=O)NCC(CN(C(=O)CCN2CCNC(=O)C2)C)O)cccc2nn[nH]c12 C1(NC(c2c(C(C)C)noc2)=O)CCCC(NC(=O)C(F)C(C)C)C1 CCCCC(O)C(C)C(=O)NC1CCCCN(C(=O)CSc2cn[nH]c2)C1 CC(C)(C(=O)NC1COCC1NC(C1(c2cncnc2)CCCC1)=O)C1CC1 Cc1cc(C(N2CCCC2C2CCN(C(C3CCCN3C3CC3)=O)C2)=O)no1 c1(OCC)cccc(C(=O)NCC(C)(C)C(=O)NCC2CCCO2)c1 CCC(C)C(O)CC(=O)N(CCC(N1CCCC(F)CC1)=O)CCCO N1(C(CSCC(=O)OC)=O)CC(NC(=O)CSCC2CCCCO2)CC1(C)C N1(C(C2CC(OC)C2)=O)CC(C)(C)C(NC(C2C=CCCC2)=O)C(C)(C)C1 N1(C(C2C(CN(C)C)C2)=O)CCC(CO)(NC(c2ccncc2O)=O)C1 C1(C(=O)NC2CCC2NC(C2CC(C(C)C)C2)=O)(CC)CCCC1O c1(C(N(OCC(=O)NCC2CN(CC)C2)C)=O)c(C)noc1C1CC1 C12(CNC(c3[nH]ccc(=N)n3)=O)CCCCC1CN(C(=O)C=C1CCCC1)C2 c1(C(N2CC=CC(NC(C(C(C)C)n3cnnc3)=O)C2)=O)ccc(Cl)c(C#N)n1 N1(CCC(=O)NCC(CNC(C(OC)OC)=O)(C)O)C(=O)NC(C)(C)C1=O Cc1nc(C(N2CCC3(CC3C(=O)N(CC(N3CCCC3)=O)CC)C2)=O)ccc1C#N Cc1cc(C(=O)NC2CCN(C(=O)C=Cc3cn(C)cn3)C(C)C2)cnc1O CC1CN(Cc2ccon2)CC1c1nc(-c2ccc(F)cc2)no1 c1(CCC)nc(C)c(C(=O)NC(CNC(C2CC(=O)N(C)C2)=O)CO)o1 c1(N(C)CC23CCC(CC2)C3)nc(N2CCC3(C)C(C2)C3(Cl)Cl)c2ncccc2n1 O=C(C1CCCc2sccc21)NCC12CCC1CN(C(=O)CCn1cncn1)C2 N1(C(C(c2ccc(C)o2)C)=O)CCCCC1CCN(C(=O)CCCN(C)C)C N1(C(C(C)CS(C)(=O)=O)=O)CCC(C2(NC(c3coc(Cl)c3)=O)CC2)CC1 C(=O)(C(CO)C(F)(F)F)NC(C(=O)N(C)Cc1ncccn1)C(C)(C)C N1(C(c2n[nH]c(C)c2Cl)=O)CC23CCCC2(C1)CN(C(C1(C)CCCCC1)=O)C3 C1(NC(CC(c2ccc(OC)cc2)NC(C)=O)=O)CCCCC(C)(C)C1 Cc1cc(C(N2CC(NC(c3cc(-c4cccs4)[nH]n3)=O)C(F)C2)=O)ccc1F CC1CC(=O)Nc2ccccc2N1C(c1cc(C(C)(C)N)no1)=O n1(CC)cc(C(N2CCC(C)(CNC(=O)C=C3CCC3)C2)=O)c(C(C)(C)C)n1 Cc1ncc(Cl)cc1CC(=O)NC(CNC(=O)CC(C)N(C)C)CC(C)C N#Cc1cc(C(N2CC3(c4ccccc4OC(F)F)CC2(CO)C3)=O)cc(O)c1 C(C(CC1CC1)C(=O)NCC=CBr)NC(CC#N)=O C1(C(N2CC(CCNC(c3c(C)[nH]cc3)=O)OCCC2)=O)CCC2(CCC2)CC1 c1(OCC)cc(F)ccc1-c1cnc(Cl)c(C(N2CC(N(C)C)C(C)(C)C2)=O)c1 c1(C(=O)NC2CCC(NC(CCNS(CC)(=O)=O)=O)CC2)cccn2cnnc12 N12CCN(C)C(C1)C(=O)NCCOC(CC)C2=O.C(CCCSC)OCC C1(CC(=O)NCC(=O)NCC(=O)OC(C)(C)C)CCCC(NC(=O)CC(F)F)C1 N1(C(C(C)NC=O)=O)CCN(C(=O)CCn2cncn2)CC1Cc1ccccc1 C1(C(N2CC(C)(C)C(CNC(C3COC3)=O)C2)=O)CC2CCCC(C1)C2 C1(N(C(c2n(CC)cnn2)=O)C)CCN(C(c2cnc(Cl)s2)=O)CC1 c1(CC)ccccc1C(=O)NCCC1CCCN(C(=O)C(C)=CCO)C1 c1(OC)ccc(NC(=O)CCCCCN(C(=O)C(C)NC(N)=O)C)c(C)c1 c1(C(=O)NCC(C)NC(C2C(CCC)C2)=O)cccc(N)c1C Cc1cc(OC(C)C)c(C2CCCC=CN2CC(O)COCC(C)C)cc1F C1(C(=O)NCC(C)NC(=O)C(=Cc2c[nH]cn2)F)CCS(=O)(=O)C(C)C1 c1(OC)ccc(F)c2[nH]c(C(=O)NCC3(NC(C4COC4)=O)CCOC3)cc12 N1(C(C2N(C)CCC2)=O)CC2(CC(NC(C3(c4cccnc4)CCC3)=O)CO2)C1 c1(C(N2C(CNC(C3N=C(C)SC3)=O)CC(O)C2)=O)cnn2c(C)ccnc12 C1(CC)(NC(=O)CC2COCCN2C)CCN(C(c2cnncc2NC)=O)CC1 c1(C(N2CC(NC(C3(C)CCCCO3)=O)C2)=O)cn2c(n1)CCCC2 C1(C(N(CCC)CCN(C)C)=O)CCC2CCC1N2C(=O)C=CC(F)(F)F n1(CC)cc(C)c(CN2CCOCC2c2cn(C3CCC3O)nn2)n1 N1(C(CC(C)P(C)(C)=O)=O)CC2OC(C)(C)OC2C1 c1(C(=O)NC2CN(c3ccnc(SCC(=O)OC)n3)C2)ccc(OC)cc1 N1(C(CC2C(C)(C)C2)=O)CCN(C(=O)CSCC(N2CCCC2)=O)CC(O)C1 CC(C)(C#N)C(=O)NCC(O)CC(=O)NCc1cccc(O)n1 CCCC(F)C(=O)NCC1(C(=O)NCC(CC)N(C)C)CCC1 N1(C(c2cc(C)cc(Cl)n2)=O)CCC2(CCCCN(C(c3ccncc3)=O)C2)C1 C#CCCN=C(NCCc1cccc(C#N)c1)NCC1CN(C(C)=O)CCO1 C1(CNC(=O)COc2cccnc2CSCc2ccccc2)CC2(CCC2)CO1 N1(C(CCN(CCC)C)=O)CCC(O)C(C(=O)NCCC(=O)OC)C1 N1(CC(=O)N(C(C)C(=O)OOCC)CCOC(C)C(=O)OC)CCCC1C.O CC1(C)CC(CC(=O)NCc2cccc(Cl)c2)CN1C(=O)Cn1cccn1 CC1OC2CCC1(NC(=O)CC1CCCN(C(=O)CC3(N(C)C)CC3)CC1)C2 c1(C(=O)NCCN(CC(C)O)C(C2C(=C)C2)=O)ccc(C(C)=O)n1C c1(C(=O)OC)cccc(C)c1S(=O)(=O)NC1CC1C(N1CC2CCC(C1)O2)=O Cc1cccc(NC(=O)C(C#N)=CCCC(=O)NOCC2CCN(C)CC2)c1C O=C(CCCCO)NCC(=O)NC1CC(F)(CNC(=O)CSC2CC3CC3C2)C1 C1(CNC(c2cc(CC)sc2)=O)CN(C(=O)CN(C(=O)C(C)C)C)CC1(C)C C12(C(=O)NC3(C)CCOCC3)CC(CN(C(=O)CC=Cc3ccccc3)C1)C2 C(=O)(CCCCCF)NC1C(CNC(C2(NS(CCCC)(=O)=O)CC2)=O)CC1 C1(COC)(NC(=O)CC(C)SC)CCCN(C(c2cnc(C3CCC3)s2)=O)C1 C(=O)(C1=CC(O)C(NC(=O)C#CC2CC2)C1)NC(c1ccccc1)C#C c1(-c2c(C(=O)NCC3(C(C)NC(C(C)=CC)=O)CC3)c[nH]c2)ccc(F)cc1 c1(C(C(=O)NCC(CNC(=O)C#CC2CC2)OC)O)cccc(F)c1 C1(C(=O)NC(CCCC)COc2ccccc2)CN(CP(C)(C)=O)C1 C1(C)(C(=O)NCC(CNC(C2(SC)CCC2)=O)C)CCCOC1 CCC(C)CC(=O)N1CC(O)CC1C(=O)NCCC1CC(C)C1 CCC(CC)C(C(=O)N(CCNC(C1CCCSC1)=O)C(C)C)OC c1(C)ccc(Cl)cc1.c1(CO)cc(C(c2nnnn2C2CC2)Nc2ccccc2)on1 C(N=c1nc(C(F)(F)F)[nH]s1)C1N(C(C(c2ccc(C)s2)C)=O)CCCC1 Cc1cc(Cl)c(C(=O)NCCCOCCN(C(=O)CC2OCCC2C)C)s1 c1(C(=O)NC(C2CCOC2)C#C)ccccc1Br.C1C(=O)N1 CCC(C)(C)CCCC(=O)NCC1CCCN1C(C1C2Cc3ccccc3C12)=O C1(C(N2CCCC3(CCC3)C2)=O)CN(C(C23CCCC2C3(F)F)=O)CC1C1CC1 C=CCCCCCC(=O)N1CC(C(=O)N(C(C)CCCC)C)CC12CCC2 N1(C(C(COC)(C)C)=O)CCC(NC(c2ccc(S(C)(=O)=O)s2)=O)C(CO)CC1 C1(C(N(CC(C)NC(C2(CF)CC2)=O)C)=O)CC2(CCCC2)CO1 c1(C(N2CCC3CCC(C2)S3)C(=O)NCCCOC)ccc(F)c2[nH]ncc12 C(=O)(C#CC1CCOCC1)NC1CN(C(C(c2cccc(C)c2)=O)=O)CC12CC2 CC(C)CCC(C(=O)NC1CNC(=O)C12CC2)NC(=O)CCC1CCCC1 Cc1cn2cccc(C(N3CCC(C(C)Nc4cc(=O)n(C)cn4)C3)=O)c2n1 C#CC1C(C(=O)NCCN(C(=O)CC2CCN(C(C)=O)CC2)C)C1(C)C c1(C(=O)OC)cnc(C(N2CCN(C(=O)CSC(F)F)CC(O)C2)=O)c(Cl)c1 CC1(C)CC(C(=O)NC2(C)CCOC2=O)N(C(C2CCC2C(C)(C)C)=O)C1 C1(C)(N(C(=O)C(N)Cc2cccnn2)C)CC2(CCC2)C1 CC1CN(C(C23CC(C(C)(C)C)(C2)C3)=O)CCCN1C(=O)C1=NOC(C)C1C C1(NC(COCCCC(C)C)=O)CCN(C(=O)Cc2ccns2)C(C2CC2)C1 c1(C(N(C(C)CN(C(=O)CNS(N)(=O)=O)C)C)=O)cnn2c1CC(C)CC2 Cc1cnc(C(=O)NCC2CC2NC(c2csc(-c3ccco3)n2)=O)cc1C#N CON1CCC(C(=O)N(C(C)CN(C)C(c2c[nH]c(=N)nc2C)=O)C)CC1 C(c1cncc(O)c1)=CC(=O)NCC(C)N(C)C(C1CC12CC(F)(F)C2)=O Cn1c(CN2C(C)CC2(C)C)cnc1Cl.C12CC(C1)C(=O)O2.C(C)(C)(C)O c1(C(=O)NCC2(C)CCC(NC(=O)C3=NNC(=O)C3)C2)csc2cccnc12 c1(CC(N2CCOCC2CNCC2CCC2)=O)ccc(Br)c(F)c1 C1(C)(CNC(CC(C)SC)=O)CCCC1NC(c1ccc(COC(C)=O)cc1)=O c1(OC)cc(CCC(N2CC3CC2CN3C(=O)C=C2CC2)=O)ccc1Cl c1(C(N2CCN(C(CSCCCC)=O)C(C)CC2)=O)cccc2c1C(C#N)C2 C(=O)(C(CNC(=O)C=Cc1nccs1)C(C)(C)C)NC(C(CC)C)CO c1(CC)nc(C(=O)NC(C)CCN(C)C(C2CCC(CN(C)C)O2)=O)cs1 c1(C(C)=O)cncc(C(=O)N(C)CC2CCCN2C(C2CCCC(=O)N2)=O)c1 Cc1nc(C(F)(F)F)c(C(=O)NC2CCN(C(c3ccnnc3)=O)C2C)o1 C(C)(C)(C(=O)NC1CC(O)(CNC(=O)CCOCC2CC2)C1)OC.C1(O)CCCO1 C1(NC(CSc2c(C)nccc2)=O)CCOC2(CCN(C(=O)CN(C)C)CC2)C1 c1(C(=O)NCC(C)N(C(CN(C(=O)OC)C)=O)C)cccn(O)c1=O C1(C(N2CC(N(C(C(C(C)C)NC(C)=O)=O)C)C2)=O)CCn2c(O)nnc2C1 c1(OC)cc(CC(=O)OCC2(c3ccccc3)COCCO2)ccn1 N1(C(=O)C(O)C(F)F)CCN(C2CCN(C(=O)C(F)(F)F)CC2)C(=O)C1 c1(C(=O)NC2(CO)CCN(C(CS(=O)(=O)NC)=O)C2)cnc2nccn2c1 Cc1cccc2c1CCN(c1ccc(S(=O)(=O)N(CC(C)CCO)C)cc1F)C2 N1(C(c2cc(C)nn2C)C(=O)Nc2ccccc2)CCOCC(C)(F)C1 C(=O)(C1=NOC(C)C1)N1C(CN(C(CC=C)=O)CC)CC(OC)C1 c1(C(=O)NCCN(C(C2(C)CC(F)(F)C2)=O)CC)ccc(-c2nnco2)cc1 c1(C(=O)NCCNC(C(CC)(C)F)=O)cc2n(n1)CC(C)NC2=O C1(N(C(CCOCCN(C(=O)C(O)CN(C)C)C)=O)C)CCN(C)C1(C)C c1(CNc2cncc(C(=O)Nc3cnc4sccc4c3)c2)cccc2c[nH]nc12 c1(SC)cccc(C(N2CCC(NC(c3ccc(Br)o3)=O)CC2)=O)c1O c1(CC)cncc(NC(=O)Nc2ccccc2C(c2ccc(CO)cn2)=O)c1 Cc1cnc(N2CCC(C)S(=O)CC2)c(S(=O)(=O)NC(C)Cc2cnc[nH]2)c1 c1(C(=O)NC2CCC=CCCC2)sc2ccccc2c1Cc1nc[nH]n1 c1(OCC)cccc(-c2nc(CCC)n(C(C)COCC)n2)c1.C(C)(C)(C)S C=CCCCCC(=O)NC1CCC1NC(c1ncoc1C(C)C)=O Cc1cc(NC(=O)CC2CC(F)(F)CN2C(=O)CC23CCCC2C3)cnc1Cl C1(CC(=O)NC)SC(=Nc2ccc(C)cc2)N(CC(N)C2CC2)C1=O c1(OC)cc(CNC2CCCC2C(N2CC3CC3C2C#N)=O)ccc1Br c1(C(N2CCOCC(NC(C(C)(C)SC)=O)C2)=O)cc2c(F)cccc2s1 CCCCCS(=O)(=O)CC(=O)NCC1CC(C)N(C(c2cc(CO)c(C)o2)=O)C1 C(CC(C)(C)CC(=O)N1CCC(C)(NC(c2c[nH]c(C(N)=O)c2)=O)CC1)OC C(=O)(C1=C(Cl)CCC1)N(C)CC1(NC(CNc2c(OCC#C)cccc2)=O)CC1 Cc1cncc(C=CC(=O)NC2CCC2NC(c2cccc(C(C)C)n2)=O)c1 C#CC1CCN(C(=O)Nc2cnn(-c3ccc(C)cc3)c2C)C1 C(=O)(CCC(=O)N(C)C)NC(C)CCNC(C1CC(CF)C1)=O c1(OCC)ccc(F)c(C(N2CCN(C(=O)COC)CC2C(C)C)=O)c1F N1(C(CCc2cc(C)ncc2)=O)CCN(Cc2cc(Br)c(C)cn2)CC1C#N C1(c2nnnn2C(C)(C)CC)(NC2CC(C=C)C2)CCCCCCCC1 N1(C(CC2C(C)CCO2)=O)CCC(NC(=O)C(F)C2CCCC2)CC1C c1(C(=O)NC2C(NC(C3CC(SC)C3)=O)C2)c(OC(F)(F)F)cccc1F N1(C(C(C2CCOCC2)OCC)=O)CCC(F)(CNC(=O)C2=CCOC2)C1 C1(C)(C(N(C(C)C(N2CCC(SCCN(C)C)C2)=O)C)=O)CC2CCC1O2 N1(C(c2cn(CC)nn2)C(=O)NCCC(=O)OCC)CCOCC12CCS(=O)(=O)C2 Cc1ccc(C(=O)NC2CN(C(C(=O)NCCCF)=O)CC2C(F)(F)F)cc1C C1(OC)CCC2(C(N3CCCC(CCNC(=O)Cc4cccs4)C3)=O)CCC12 c1(NC(C2CCN2C2CCCC2)=O)cccc(CC2(CO)CCCC2)c1 c1(C(N2CCCC(C(C)NC(c3c(C)nc(C)s3)=O)C2)=O)ccn2cncc2c1 c1(NC(=O)C=C2CCN(C(=O)CCCC3CC3)CC2)cncc2ccccc12 N1(C(C(=O)NC(C)Cc2ncon2)C)CCCCC1=O C1(CC=C)(NC(c2cn[nH]c2)=O)CCN(C(C2CCCC2c2cnn(C)c2)=O)C1 C1(C(N2CCCCC(CNC(CC(=O)NC3CC3)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 c1(C2C(NC(C3C(n4cc(C(C)O)nn4)CCCC3)=O)C2)ccc(F)cc1Cl c1(C(N2CC(F)(CNC(c3scc(OC)c3)=O)C2)=O)sc(F)cc1Cl C=C(C)C1OCCC1CNC(=O)CC(C)CNC(c1csc(C)n1)=O c1(C(C(=O)NC(C)CC)N(C2CCCCC2)CC=C)sc(Cl)cc1Br N1(C(Cc2cn(C(C)C)nc2)=O)CCC(CNC(=O)C(F)(F)C(C)O)C12CC2 c1(C2c3nnnn3CCN2)cc2cc(Br)ccc2o1.C1(CC=C)(OCC)CCC1 CC(C)(F)CCC(=O)NC(C1CCCCC1)CNC(=O)CC=C(Cl)Cl c1(C(=O)NCCN(C(=O)CCC2OCCO2)CCC)sccc1Cl C12(NC(CC(C)SC)=O)CCOC(CNC(c3cncn(C)c3=O)=O)(C1)C2 c1(C(=O)NC2(NC(C(C)OCCOCC)=O)CSC2)cccc(O)n1 C1(C(=O)NC2CC(CNC(C=C3CCN(C)C3)=O)C2)CCC2(CCCCC2)C1 c1(C(=O)NCC2C(NC(c3cc(F)ccc3F)=O)CCC2)csc2c1CCCC2 c1(C(=O)NCC(CNC(CC(C)C)=O)(C)O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 c1(C(C)NC(N(CC(C)C#N)CC)=O)csc(C)n1 N1(C(C(CC)F)=O)CCN2CC1C2=O.c1(C(=O)OC)ncc(C(F)(F)F)cc1Cl c1(C(C)C)cccc(C(=O)NC2CC(F)(CNC(c3nc(=O)n(C)[nH]3)=O)C2)c1F C12(NC(CCNS(CC)(=O)=O)=O)CCCC(CN(C(C3CC4CCC4C3)=O)C1)C2 N1(C(Cn2ncc(C#N)c2)=O)C(C(=O)N(CC2CCC2)CC2CC2)CCC12CC2 N1(C(CC(CNC(c2ccn(C)c2)=O)OC)=O)CCOC2COCC2C1 Cc1nc(N(CC(C)C#N)C)cc(NC2CCN(CC3CC3)CC2)n1 C1(CC)CN(C(c2ncc(C)cc2Br)=O)CCN1C(=O)C(C)C(O)CC C1(C(N2CCN(C)C(CNC(=O)CCC(F)F)C2)=O)CC2CCC1C21CC1 n1(CCC)ncnc1CN(CCNC(=O)C(C)C1CC1)CCOC CN1CCN(C(C2(C3CCCN3C(=O)CCc3cnoc3)CC2)=O)CC1=O N1(C(c2c(F)ccc(C)n2)=O)CC2CCN(C(=O)C=Cc3cncc(O)c3)C2C1 C(=O)(C(C(=O)NCC(C)N(C)C(C12CC(C)(CO1)C2)=O)C(C)C)OCC CC(C)CC(C)CC(=O)N1CCC(C(=O)NCc2ncnn2C(C)C)O1 CC1CCOC1C(=O)NC(C1CCCCC1)C(=O)NC(C)Cc1cn[nH]c1 CC1(C)CCC(CO)N(C(C2(NC(C3CCSC3)=O)CCOCC2)=O)C1 c1(OCC)cc(C(=O)Nc2c(F)ccc(F)c2O)ncc1C1=COCCC1 C1(NCc2conc2)CCN(C(=O)NC)CC1.C#CCOCC1CC1 C1(C(=O)NCCNC(C2CCCCC2)=O)CN(C(=O)CC2CC2)C2(CCC2)C1 C1(C(N(C2(CC)CC2)C)=O)CN(C(c2scc(C)c2C)=O)C(C)(C)C1 c1(C(N2CCC(C3N(Cc4nnc(C)o4)CCC3)CC2)C)cnn2c1CCCC2 N1(c2ccnc(NC3CC(C)C3)n2)CCCC2CCCCC12 C12(NC(C(C)n3ccnn3)=O)CCCCCC1N(C(=O)C=CC=C(Cl)Cl)CC2 CCC(CCC(=O)NCC(c1cccc(Cl)c1)NC(=O)C=Cc1cc[nH]n1)OC c1(C(N(CC(CNC(C(CC)NC(N)=O)=O)C)C)=O)ccc(C)nn1 CCCC(CCCO)C(=O)NC1CCN(C(=O)CCc2ccc(N)cn2)C(C)C1 C1(C(=O)OCC2C(C)C2)COCC1NC(=O)OC(C)(C)C C(=O)(CC(O)C(C)CC)NCCCC(=O)NCC(CC)(F)CC N1(C(c2c(OCC)ccs2)=O)CCC2(CCN(C(C3CCC(=O)O3)=O)C2)C1 n1(C(C)OC)c(CCNC(=O)NNC(=O)C(F)c2ccccc2)nc2ccccc12 C1(C(=O)NCC(C)(O)C2CCCC2)CCN(C(=O)C2(F)CCCCC2)O1 C1(C(=O)NCC(C)CNC(c2cnc(C(F)(F)F)s2)=O)CC(=O)N(C)C1 N1(CC)CCC(CNC(c2ccc(OCCN)cc2)=O)C(C)C1 C1(CC(C)NC(C2N(C(C)=O)CCC2)=O)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 C1(NC(c2cc(C)oc2)=O)CCCN(C(c2cccc(C)c2Cl)=O)C1C Cc1ccc(C(=O)NCC2CC(NC(C3CCC3(C)C)=O)C2)cc1O C12(C(N(C3CCCN(C(C4CCCCS4)=O)CC3)C)=O)CC(C)(CCO1)C2 c1(OC)ccccc1C(O)C(=O)NCC1(C)CC(NC(=O)Cc2cn(C)cn2)C1 C1(NC(Cc2ccc(OCC)cn2)=O)CC(O)CN(C(c2ccncc2Cl)=O)C1 c1(C(N2CC(C(=O)NC(CC)C(C)C)OC(C)C2)=O)cc2ccccc2[nH]1 CN1CC=C(CC(=O)NC23CC(C2)N(C(C24CCCC2C4(F)F)=O)C3)CC1 C1(NC(=O)CCc2cccs2)CC2CCC1N(c1ncncc1Cl)C2 N1(C(c2c(CCC)occ2)=O)CCCCC(CNC(c2ocnc2C2CC2)=O)C1 C1(OC(C)=O)CCN(C(c2cc(CNC(C3CC3F)=O)cs2)=O)C1 c1(C(N2C(C(N3CCCC3c3ccccc3Cl)=O)CC2)=O)cc[n+]([O-])cc1 CC1CCN(C(C2CC2F)=O)CC1NC(c1cccc(-c2nc[nH]n2)c1)=O C(=O)(CC(C)(C)CCOC)NCC1C(CNC(C(CC=C)C)=O)C1 C(=O)(C(C)C(C)C(C)(C)C)N(CCN(C(C(CC=C)C(C)C)=O)C(C)C)C C1(NC(COCCC=C)=O)CN(C(=O)CNc2nccs2)CC12CC2 C(=O)(N=c1[nH][nH]c(C)c1C)c1c(C)nc(NC(c2ccc3cc[nH]c3c2Br)=O)s1 C1(OC)CC(F)CN(C(c2c[nH]nc2CNC(=O)CCc2nc[nH]n2)=O)C1 c1(C(C)C)ccc2c(c1)CCN(C(c1cccc(Br)c1Cl)C(=O)NC1CC1)CC2 O=C1CCC(C(=O)N2CCCC2C(C)NC(c2nccn3nccc23)=O)=NN1 N1(C(C(CC)SC)=O)CC2(CCN(C(=O)CCc3nc(C4CCC4)no3)CC2)C1 C(=O)(CC1=CCOCC1)NC(C1CN(C(C(C)n2ccnc2)=O)C1)C N1(C(C=Cc2cn(C)nn2)=O)CCC2(CCN(C(C3CC(O)C(F)C3)=O)CC2)C1 c1(CNC(CCNC(C2(CC)CCCC2)=O)=O)cccc(Cl)n1 c1(C(C)=O)ccc(C(=O)N(C2CCN(CC(O)COCCC(C)C)C2)C)s1 C1(C(N2CCC(O)(C(C)C)C2)=O)CC2(CCN1C(c1ccnn1C)=O)CC2 C(C(C)(C)CC(=O)NCc1nc(C)cc(O)n1)NC(c1c(CC)nns1)=O c1(OCC=C)c(OC)cc(COc2ccccc2N2CCC(O)CC2)cc1Cl C(=O)(C(C)(C)c1ccn(C)n1)NCCN(C(=O)CC1CCC1(F)F)CC n1(CC(=O)NCC(CNC(CCc2cc(C)n(C)n2)=O)F)cccc(N)c1=O c1(C(=O)NCC2(O)CN(C(C(CC)(C)C)=O)C2)nccc(Cl)c1Cl C(=O)(C1=C(Cl)CCC1)NC(C(=O)NC1(C)CC1(F)F)C1CCCO1 N1(C(c2ccno2)=O)CCCC2(CCCCN2C(c2c(Cl)cncc2Cl)=O)C1 C1(C(=O)NCC2N(C(CCCC#C)=O)CCCC2)CCC12CCCC2 C1(F)(CNC(CCC2(C)CC2)=O)CCN(C(C2COCCO2)=O)C1 C1(NC(c2n(C)nc(O)c2)=O)CN(C(=O)CN2CC3CC3C2)C2CCCC12 C1(NC(=O)CC2CC3(CC3)C2)COC2(CCN(C(=O)C#CC3CC3)CC2)C1 c1(NC(c2nn(C)cc2NC(C)=O)c2n(CC(=C)C)nnn2)cccc(OCC)c1 Cc1ccc(N)c(C(=O)NCC(C)(C2CC2)NC(c2csc3nnsc23)=O)c1 c1(C(=O)NCCCCC(C)NC(C2CC2(C)C(F)(F)F)=O)ccc2c(c1)OCC2 N1(C(C(C=C=C)C)=O)CCC(C2OCCO2)CC1NC(=O)CCCC(F)F c1(NNC(C2CN(C3COC3)C2)=O)ccc(C2COC2)cc1F.C12CCN(C1)C2 N1(C(c2c(CC)ccs2)=O)CCN(C(=O)CC2CCCCC2)C(C)C1 C1(NCCCC(=O)NCc2ccc(C#N)cc2)CCn2ccnc2C1 c1(C(=O)OC)ccc(C(=O)N(C)CC2CN(C(c3ccccn3)=O)C2)cc1C C1(C(C)NC(=O)C(F)Cc2ccccc2)CCCN(C(=O)C(Cl)=CCl)C1 C1(C(=O)NC(CNC(c2ccn(C(C)C)n2)=O)C2CCC2)CN2CCN1CC2C Cc1cccc(NC(=O)CN2CCC(NC(=O)Cc3nocc3C)CC2)c1 C#Cc1ccc(F)c(C(N2CCCC2CN(C(=O)CCC#CC)CC)=O)c1 Cc1ccc(C2(C(=O)OCCC3CC(C(F)(F)F)C3)CCCC2)cc1 c1(C(N2C(C(C)NC(CN(C3CC3)CC)=O)CCC2)=O)ccc([N+](=O)[O-])c(N)n1 C(=O)(C(C)C(C)CC)NCC(CN(C(C1(CCC)CC1)=O)CC)(C)C n1(CCC(=O)NCCC(=C)CNC(=O)CCC2CC2C)ccc2cc(Cl)ccc12 N=S1(=O)CCC(NC(C2(O)CCCNC2)=O)c2cc(F)ccc21 c1(C(=O)NCC=CCNC(c2cnsc2)=O)cccc2[nH]ncc12 N1(C(c2c(SCC)ccc(Cl)c2)=O)CC2CC(NC(=O)C(C3CC3)OC)CC2C1 Cc1cn(C)cc1C(N1CC(O)CC1CNC(=O)C(c1ccccc1)=O)=O N1(C(C2CC(OC)C(OC)C2)=O)CCCC(C2CCN(C(=O)CNC(C)=O)C2)C1 c1(NC(C2CC2(c2cc(F)cc(F)c2)F)=O)cnc2cnccc2c1 CC1(CNC(C2CC(=C3CCC3)C2)=O)CN(C(C2CCCC2)=O)CCO1 c1(N2CCC(C(C)NC(=O)C(C)(C)C(F)F)C2)nc(Cl)ncc1[N+](=O)[O-] C1(CCC(=O)NCC2CC(F)(CNC(Cc3ncn(C)c3)=O)C2)CCCC(=O)N1 CC1CC(CC(=O)NC2CCN(C)CC2)CN1C(c1ccc(N)cn1)=O N1(C(C(C)OCC#C)=O)CCCC12CCN(C(=O)CSC1CCOC1=O)CC2 C12(C)CCCN(C1)C2=O.C1(CC(=O)NCC)CC(C)=NO1 C1(CC#C)(C(=O)N(CCCC(=O)NCCCCSC(F)F)C)CCCCC1 Nc1ccc(F)cc1C(=O)NCC1CCCCC1NC(=O)Cc1ccc(F)cc1 CC1CN(C(C2CC(N(C)C)C2)=O)CCC1C(=O)NC1CCN(C2CC2)CC1 C1(NC(C2C=CCC2)=O)COC2CN(C(c3ccc(-c4ccccn4)o3)=O)CC12 N1(C(c2c(OC)ccs2)=O)CCCC(C)(NC(c2ccn(C(F)(F)F)n2)=O)C1 C1(NC(C2CC(C(C)C)C2)=O)COC2(C1)CN(C(C1CC(C)OC1C)=O)C2 c1(CC(=O)NCC(C)(CO)NC(c2ccc(COC)[nH]2)=O)ccnc(C(N)=O)c1 C1(NC(C(C)(C)OCC)=O)CCC(C)(NC(=O)CSc2ccncc2)C1 C(CCC(C)C(=O)NCCC1CC1C(N1CC(CO)C1)=O)OC Cc1cccc2c1OC(C(N1CC3C(NC(C4(O)CCCCCC4)=O)C3C1)=O)C2 c1(OC)ncnc(C)c1C(N1CC2C(NC(=O)CC(C)n3ccc(C)n3)C2C1)=O CC1(C2(C)CN(C(=O)CN3CCOC3=O)C2)CC2(CC2)C1.C12CCCC1C(=O)NC2 C1(NC(c2nnc(C)s2)=O)CN(C(=O)C(C)O)C2CCCCC12 c1(C(=O)NC(C)C(C2CCCCC2)NC(=O)Cc2cnns2)cc2sccc2[nH]1 C(=O)(CCC(=O)NN(C)C)N1C(C(C)C)CN(C(C)=O)CC1 C=CC(C)(CC)C(=O)N1CCC(C(=O)Nc2cccc(O)c2F)O1 CC(CC(=O)NCC(C)CNC(=O)CCN1C(=O)CCC1=O)CC(F)(F)F N#Cc1ccc(C(N2CC(NC(c3ccncn3)=O)C(F)C2)=O)cc1Cl N1(CC)CCCC1C(=O)NCC1CC1CNC(c1scnc1C(F)(F)F)=O N1(C(c2c(C)snn2)=O)CCC2(CCCN2C(C2CCN(CC(C)C)C2)=O)CC1 N1(c2nnc(CC)n2CC2CCCC(C)C2)CCC(S(=O)(=O)CC)CC1 C123CCC(CO1)(C2)C(=O)OC3=O.CCC(C)CC(=O)N(CCN1CCCC1)CC c1(OC)nccc(C(=O)NC2C3CN(C(c4nn(C)nc4C)=O)CC23)c1F C(=O)(CS(F)(F)(F)(F)F)N1C(C)CCCCC1 C1(C(=O)NCC(C(C)C)NC(C23CC4CC2C3C4)=O)Cc2ccc(F)cc2O1 C#CCCCCC(=O)NCC1CCCC1NC(C1(F)CCN(C)CC1)=O C1(C(=O)NC(CNC(C=C(CC)C)=O)C2CC2)(OCC)CCOCC1 c1(CC(C)C(=O)N(CCCNC(C2CCCN2C)=O)C)ccccc1F C1(NCc2c(N(C)C)ccs2)CCN(C(c2cc(F)nc(F)c2)=O)CC1F CC1CCC(NC(c2c(F)cncc2Cl)=O)CN1C(c1ccnn1C)=O CC1CN(C(=O)CCc2cnn[nH]2)CCN1C(=O)COc1cccc(F)c1 Cc1ccc(=NCCC(=O)NCC(O)CNC(C2CC(C(F)F)C2)=O)[nH]c1 Brc1cc2n(n1)CCN(Cc1cc3ncccn3n1)C2 N1(CC)CCOCC1C(N1CC(C(O)C(=O)NCc2cc(OC)no2)C1)=O.C1(C)CC1 C#Cc1cnc(C(N2CCCCC2C(=O)NCC)=O)c(C)c1.C(CO)(CC(F)(F)F)N N#Cc1c(F)c(NC(c2cnn(Cc3ccccc3Cl)c2)C(F)F)cc(F)c1F N1(C(Cn2cnc(=N)[nH]2)=O)CCOC(CNC(c2cccnc2)=O)C1 c12ccc3nc(oc3c1)N1CCN(CC1CC(F)F)C2=O.C=C1CC1C(=O)OC c1(OC)ccccc1-n1cc(CN2CCC(C(C)OC(C)C)(CSC)C2)cn1 c1(NC(C2C(C)(CC)C2)=O)cnc(-c2ncccn2)s1.C12CC(C1)CNC2=O N12CC(CC13CCC3)C2.C(=O)(C(C)n1cccn1)NCC.C(C=O)OCCOCC c1(C(=O)NCC2CCN2C(c2cnns2)=O)cc(Cl)ccc1Cl C1(C(=O)NCC(C)NCc2nc[nH]n2)CCC(Cc2cnn(CC(C)(C)O)c2)CC1 S(=O)(=O)(c1cccc(Cl)c1F)N1C2CCN(S(CC(=O)OCC)(=O)=O)CC2CC1 C1(NC(C(CC)C)=O)(CNC(=O)CNC(=O)CCCCO)CCCCC1 c1(C(=O)NCC2N(C(C3C(C)C3)=O)CCC2)cc(O)c2cc(F)cc(F)c2n1 Cc1c(C(N2CCC3(CC3C(=O)Nc3cncs3)C2)=O)cccc1C(F)(F)F C1(C(C(=O)N(C2CCN(C(c3sccc3Cl)=O)C2)CCC)O)CCOCC1 N1(C(C(=O)NCCC(=O)OCC)C2CC2C2OCCO2)CCCC2(C1)OCC1CC21 C1(CNC(CC=C=C)=O)CN(C(=O)COc2nc(O)nc(O)n2)CC12CC2 N1(CC)CCN(C(=O)CC2C3CCCC3N2C(=O)Cc2ccn(C)c2)CC1C N1(CCC)CCC(C(=O)NCC2CCCC2NC(=O)CCN(C)C(C)=O)CC1 C1(C(=O)NCC2C(N(C)C)COC2)CC(O)CN1C(C1C2CCC(F)C12)=O C1(C(=O)NCC(C)CN2CCCC2)COC2(C1)CN(C(=O)CCc1ccoc1)C2 C(C(C)CC(=O)N1CCC1CNC(C1C2CCC1(c1cccnc1)C2)=O)OC c1(CNC(C(C)N(C(=O)CCSc2cn(C)nn2)CC)=O)n[nH]c2ccccc12 N1(C(C(F)OC)=O)CC(NC(c2cc(N)ccc2O)=O)CC12CCOCC2 C1(CNC(C2(C(N(C)C)=O)CC2)=O)CCN(C(=O)C=Cc2ccco2)CC1O CC1CN(C(=O)CCCC2CCCCC2)CCC1CNC(=O)CC1(C)CC1 C=CC(C)(C)CC(=O)N1CCC(NC(=O)C(c2cccc(C)c2)C)C12CC2 N1(C(Cc2nc(C)oc2)=O)CCCC(NC(=O)C(C)C(C)(F)F)C1C c1(NC(C2C=CCN2Cc2cc(Br)c(F)cc2F)=O)cccc2ncc(Br)cc12 c1cc2[nH]c(=NCC3CCCN3CC(F)(F)F)[nH]c(=NC3CCCC3)c2[nH]1 C(C(C)(C)CC(=O)N(C)Cc1nc[nH]n1)NC(C(c1ccoc1)SC)=O C1(C#C)(C(=O)NCC(C#C)CC2CC2)CN(C(C2CNC(=O)N2)=O)C1 N1(C(c2nc(CC)oc2)=O)CCCC(CC(=O)N(C(C)CO)CC2CCC2)CC1 Fc1cc(N2CC(CNc3nccc(I)n3)OC2=O)ccc1Cl N1(C(CC(CC)OC)=O)CC(CNC(c2scnc2C2CC2)=O)C2(CC2)C1 CC1CC(CN(CCCNC(=O)C(C)(C)n2ccc(C(F)(F)F)n2)C)CCO1 C1(CN(C(C(C(C)C)F)=O)C2CC2)CCC(C)N(C(=O)CCc2ccncc2)C1 C1(NC(C(CCCN(C)C)N(C)C)=O)COc2ccccc2C1 c1(C(=O)NC)cccc(C(=O)NCC#CCNC(=O)CC2CCCC(O)C2)n1 N1(C(CC=CC)=O)CCN(C(c2cccc(CCN(C)C)c2)=O)C(CCO)C1 N(C(=NCC(F)F)N1CCC(O)CC(C)(C)C1)Cc1snc(C(C)(C)C)n1 N1(C(C2C(C(=O)O)C3CCC23)=O)CC2CCC(COC(=O)OC(C)(C)C)CC2C1 C(=O)(CC(O)C(C)CC)NC(C(=O)NCc1cnc(CC)s1)C1CC1 C12(CNC(c3ncsc3Br)=O)CC1CN(C(=O)CC1(C(F)F)CC1)C2 Cn1cc(C(=O)NC2CC(NC(=O)C(c3cccc(Cl)c3)O)C2)n(C)c1=O C=C(C)CC(C(=O)NCC1(O)CCCCCC1)NC(c1cccc(CC)n1)=O CC1(C)CC(NC(C2(O)CCCCC2)=O)CN1C(c1c[nH]cc1Br)=O c1(C(N(CC(C)NC(c2cc(O)n(C)n2)=O)CC)=O)cc(C)c(F)cn1 c1(C(=O)NC2CCCC(CNC(C=C(C)C(F)F)=O)C2)ccc2c(c1)N(C)CC2 Cc1cnc2nc(=NC(=O)NCC(N)C3CC3)[nH]n2c1 N1(C(=O)CCF)CCN(C(=O)CC2CCCCC23CC3)C(c2cn[nH]c2)C1 c1(C(=O)NCC(CN(C(c2cnc(N(C)C)nc2)=O)C)O)ccc2[nH]ccc2n1 N1(C(c2cc(-c3c(F)cccc3F)[nH]n2)=O)CCN(C(C2CCO2)=O)C(CO)C1 C(C(CC(C)C)C(=O)NCCCNC(C1CN(C(C)C)C1)=O)OC c1(C(=O)NCC2(NC(C3CC4CC4C3)=O)CCCCC2)cnc2ncccc2c1 Cc1ccc(C(N)=O)cc1C(=O)N(C)CCNC(=O)C(C)Cc1c(C)n[nH]c1C c12cccc(c1)CN1CC(OCC1)CC(=O)C2=O.C1(C2CC2)(CN)CC1.C(F)(F)F C1(NC(C(C)NS(C)(=O)=O)=O)CC2CN(C(c3cccc(C(C)(F)F)c3)=O)CC12 C1(CNC(CC=C)=O)C2CN(C(=O)C(C(C)C)c3ccncc3)CC12 N1(C(C2(C(C)C)CNC(=O)C2)=O)CCCC(CC(=O)NCC2CC2)CC1 C1(C(N2CCC(NC(C(C(C)C)N3CCCCC3)=O)CC2)=O)CCC(=O)NC1=O C1(N(c2c(OC)nc(Br)cn2)C(c2coc(C)n2)=O)CC2(CCNCC2)C1 N1(C(C(C2CCCC2)OCC)=O)CCN(C(=O)C(C)(C)CCSC)CC1CC c1(C(=O)NCC2N(C(C3CCCC(C)C3)=O)CCC2)ncnc2c1ncn2C1CC1 c1(C(c2nnnn2CC2CCC2)CCCNCC(CO)C2CCC2)ccc(Cl)cn1 C1(CNC(Cc2n(C)ccn2)=O)N(C(=O)CC(C)(C)C#N)CCC1(C)C c1(C(N2CCC(C(C)NC(=O)CCn3ccnn3)C2)=O)ncn2cccnc12 C1(C2CCN(C(C3(C(F)F)CC3)=O)CC2)(NC(c2c(C)[nH]cc2)=O)CCC1 Cc1cc2cc(C(=O)OCC3CCCS(=O)(=O)C3)ccc2cn1 C=C(C)CC(C(=O)N(C)CCNC(=O)C(C)C)NC(c1ccsc1C)=O c1(C(C(=O)NCC(C)N(C(=O)Cc2nocc2C)CC)C)ccc(F)c(Cl)c1 N1(C(C2N(C)CCN(C(c3c(CC)c[nH]c3)=O)C2)=O)CCC(F)(F)C(F)C1 N1(CC(CO)NC(C(CC)OC)=O)CCN(C(c2ccc[nH]2)=O)CC1 c1(C(=O)NCC2N(C(C(CC)F)=O)CC2)cnc2sc(C)cn12 c1(C(N(C)CC2CCN(C(C(C)n3cccn3)=O)C2)=O)cc2c(nn1)CCC2 CC(CC(=O)NC1CC(N(C)C(C2CCCO2)=O)C1)N(C)C c1(Cn2cc(C3(NC(c4ncn(C(C)C)c4)=O)CCOC3)nn2)cccc(Cl)c1 C(=O)(CCCCc1ccc(OC(=O)C(C)NC)cc1)NC(C)C C(=O)(CCCCC(C)=O)NCC1(C(=O)NCC(C(C)C)OC)CC=CC1 C(N=c1[nH]cnc(NCCCOc2ncccn2)c1C)c1c(C)nc(C)nc1O N1(C(c2c(CC)onc2)=O)C2CCC1C(CNC(c1cc(OC)ccc1N)=O)C2 Cc1cc2ccc(C(N3CCC4(CCC(NC(=O)C5=CC(C)C5)C4)C3)=O)cn2c1 Cc1cc(C)c2nc(N3CCCC(CN(C(=O)CSCC(N)=O)C)C3)sc2c1 C1(CC(=O)NC(C2CCN(c3ncc(C(C)(C)O)cn3)C2)C)CCCNC(=O)C1 c1(NC(N2CCC(C(N3CC(C)N(C)CC3)=O)C2)=O)cccc2ccccc12 N1(C(CC2CC(=O)OC2)=O)CC2CC1CN2C(=O)CCOC1CCCC1 CC1CN(C(=O)C(c2ccccc2)O)CC1NC(C1(CO)CCOCC1)=O c1(NC(c2cccc(CC)c2)=O)ncc(-c2cccc(OCC(=O)O)c2)cc1F c1(C(N2CC(C(C)NC(=O)C(O)C3CC3)C2)=O)ccn2ccccc12 C(=O)(C(O)CC(F)F)N(C1CCCN(C(=O)CC2CCOC2)CC1)C C1(C(C)C)CCCCCN1C(C1(F)CCN(C(C2CC(=O)CC(=O)N2)=O)C1)=O N1(CCC)CCCC(C(=O)NC(CNC(=O)CCc2cnc(C)s2)C(C)C)C1 CCC(C)C(C(N)=O)NC(c1csc(CNC(=O)C=CC2CCC2)c1)=O Cc1cc(Br)cc(C(=O)NC2CC(NC(c3c(Cl)cccc3I)=O)C2)c1O C(=O)(C1=CC2CCCC12)N(CCNC(c1n(CC=C)ccc1)=O)C(C)C C1(C(=O)NCC(C)NC(C2(C3CCOCC3)CC2)=O)COC2(CCC2)CO1 Cc1cnc(C(=O)NC(C)(C)C(=O)N(CC(C)O)C)cn1 c1(C(N2CCC(C)(CCNC(CCN(CCC)C)=O)C2)=O)c(F)ccc(C)c1F c1(C(=O)NC(C(C(=O)NC2(CC=C)CC=CCC2)C)C)cn(C)c(=O)cn1 C1(CN(C(C=C(C)C(C)C)=O)C)CCCN1C(c1nc(Br)c[nH]1)=O C(N=c1[nH]c(=NCC2(CO)CC23CCC3)c2sccc2[nH]1)C1(C)CCOC1 c1(OC)cc(C(=O)NC2CCCCC2CNC(C2(C(C)(C)O)CC2)=O)ccc1C C1(C)(CNC(c2nc(CCC)sc2)=O)CCN(c2nc(C(F)(F)F)ns2)C1 c1(CC)c(C(=O)N(CC(C)N(C(=O)C(C)n2cccc2)C)C)cccc1C c1(OC)cc(O)c(C(=O)Nc2cc(-c3ccco3)cc(SC(F)(F)F)c2)cc1OC N1(C(CCCCC=CC)=O)CC(C(=O)NC(C)CN(C)C)CC(C)(C)C1 N1(CCCC(=O)N(C2CCN(C(C3CC3(C)C)=O)CC2)C)C(=O)NC(C)(C)C1=O N1(C(c2n(CC)ccc2)=O)CC(F)CC1CNC(=O)Cc1cnccc1Cl N1(CCC)C(=O)NC2(CCN(C(c3cc4cnc(C)nc4nc3C)C)CC2)C1=O c1(C(=O)NCCC2OCCN(C(C(CSC)O)=O)C2)ccc(O)cc1C N1(C(C(C=C=C)C)=O)CCN(C(c2ocnc2C2CC2)=O)CC1C(F)F N1(C(c2nncc(OC)c2)=O)CCN(C(c2ccoc2C2CC2)=O)C(C)C1 C(=O)(C(O)C(C(C)C)OC)NC1CC(CC(=O)NC(C2(C)CCC3CC3C2)C)C1 Cc1nn(C)c(C)c1CNC(=O)C(CO)NC(c1ccc(F)s1)=O c1(C(=O)NCC2(CNC(=O)CCOCC(F)F)CC2(F)F)cnc(O)c(F)c1 CC1(C)CC(=O)C(N(C2CC2)Cc2cn(CC(=O)O)c(=O)nc2O)C(C)(C)C1 c1(CC(=O)NC2C(NC(c3ccc(CC)cn3)=O)CCC2)cn2cc(C)sc2n1 N1(C(CN2CC(=O)NC2=O)=O)CCOC2CN(C(C3CCCC3(F)F)=O)CC12 CC1(C)CN(C(=O)C=CCN2CCOCC2)CC1CNC(C1SCCCS1)=O c1(C(=O)NC(CN(C(C(C)OC(C)(C)C)=O)C)(C)C)ncnc2cc[nH]c12 c1(C(=O)NCC2CC23CCCC3)nc2cccc(Br)c2[nH]1 c1(C(=O)NCCN(C(C)=O)CC)cc(C#N)[nH]c1C.C12CN(C1)C(=O)N(C)C2 c1(OC)ccc(F)c(C(=O)NCC2(C)CC(NC(c3cc(CO)[nH]n3)=O)C2)c1F C(=O)(C(C(C)C)c1ccc(Cl)cc1)NC(CN(C(c1cc(C)sn1)=O)CC)C CC(C(=O)N(C1CCCC1)CCN)S(=O)(=O)C1CCOCC1 C1(CC)CN(C(=O)C(C)n2cncn2)CCC1NC(c1cccc(Cl)n1)=O Cc1ccnc(F)c1C(=O)NCCN(c1ccccc1C#N)C c1(OC)ccc2c(c1)CC(C(=O)NCC1C3CN(C(=O)CNC=O)CC13)CC2 N1(C(C2CC23CCC3)C(=O)NC(C(=O)OC)C)CC(C)(C)OC2(CCOC2)C1 C1(CC)CCN(C(C23CCC(CC2NC(c2cccc(F)c2C)=O)C3)=O)CCO1 Cc1nc2ccc(C(=O)N(C3CC3)Cc3cn(CC4CC5CC5C4)nn3)cn2n1 Cc1ccc(C(N2CC(N(C(=O)CC(C)n3cccn3)C)C2)=O)c(O)c1C N1(C(c2nnc(CC)s2)=O)CCC(NC(C2CCC(F)(F)CC2)=O)C(CO)CC1 N1(C(C=C2C(C)(C)CCCC2)=O)CCc2ccc(Br)cc2C1C(F)(F)F Cc1cc(-c2cn(C3CCC(C(=O)NCc4cccc(F)c4Cl)C3)nn2)cc(Cl)c1 N1(Cc2ccc(CC(C)C)s2)CCC(C(C(F)(F)F)NC(=O)CO)CC1 C1(CC)CCN(C(C2CCN(CC)C2)=O)C1C(=O)NOCC1CCOC1 c1(CC)occc1C(=O)NCC1CCC(NC(=O)CCSCc2ccccc2)C1 C1(O)(C(N2CCN(C(=O)CC3CC3)CC2c2ccncc2)=O)CN2CCC1CC2 c1(C2C(NC(C(CNC(CC(C)C)=O)N(C)C)=O)C2)cccc(F)c1 S(=O)(=O)(c1ccc(Br)cc1)N1C(NC(C(=O)OC)CC(C)SC)CCCCC1 c1(OC)c(C)cc(C(N2CCC(CNC(=O)CCCC#N)C(F)(F)C2)=O)cc1C S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(CNC(c2ncc(C)nc2)=O)CC1 CCC(C(C)C)NC(=O)NC(c1n[nH]c(C)n1)Cc1ccccc1 C=CC1(C(N2CC(C)(C)C2COC)=O)CCN(C(=O)CC2CCOC2(C)C)CC1 CC1(C(=O)NC2CCCC2CF)CCCN1C(c1ccc(O)cn1)=O C1(F)(CNC(CCC(=O)NC)=O)CCN(C(=O)C(c2ccccc2)C)CC1 CC(C)C(F)(F)CC(=O)N1CCN(C(C2(C)CCCCO2)=O)CC1C1CCCC1 C1(N(C(C2C(=C)C2)=O)C)CCCCN(C(=O)Cc2cncn2C2CC2)C1 c1(C(=O)NC(C)CCCNC(=O)Cc2cn(C)nn2)cc2c(O)ncnc2cn1 N1(C(Cn2c(C)nnn2)=O)CC2CC1CN(C(=O)C=CC(F)(F)F)C2 CC(C=C(Cl)Cl)C(=O)NCNc1cc(Br)c(Cl)n1C C1(C(N(C)CC2CC(=C)C2)=O)(NC(=O)CN2CCCCCC2)CCCC1C CC1CN(C(C2CCC(C3CC3)N2C(C2CCC(C)(C)C2)=O)=O)CCS1=O Cc1cccc(CC(C)NC(C(F)F)C2CCC2)c1 N1(C(C(C2CCCCC2)OC)=O)CC(O)CC1CNC(C1(CCF)CCC1)=O C1(C(N2C3(CN(C(c4cccc(=S)n4O)=O)C3)CC2)=O)CCn2ncnc2C1 c1(C(=O)NCC2(CNC(C3CC4C=CC3O4)=O)CC2)cc2n(n1)CCCO2 Cc1cc(C(=O)NCc2nocc2C(=O)NC(C23CC(CO2)C3)C)n[nH]1 N#Cc1ccccc1CC(N1CCCC1CC(N1CCOC2CC12)=O)=O N1(C(CC2(COCC)CC2)=O)C2CCC1CC(NC(=O)C(CC)CC(F)F)C2 C1(C(N(CC(C)C#N)C)=O)CN(C(c2csc(F)c2)=O)CCC1(C)C c1(C(=O)NCCCC2OCCN(C(CC(=C)C)=O)C2)cc([N+](=O)[O-])oc1C c1(C(N2C(CCNC(C3(COC)CCCO3)=O)CCC2)=O)csc2nccn12 Cc1ccc2cc(C(=O)NCCN(C(=O)C(N3CCOC3=O)C)C3CC3)cn2c1 C(=O)(CC(C)(C)C(C)(F)F)NC1CCN(C(C2ON=C(C(C)(C)C)C2)=O)CC1F CC(O)CCCCCC(=O)N1CC(NC(=O)CCc2cncn2C)CC12CCC2 Cn1nc2cc1CO2.C1(C(=O)N(C)C)CN(C(C23CCCCC2C3)=O)CCO1 c1(N2CCC(COC)C2)nc(=NC(C)C2CCCC2)[nH]c2c1CSC2 C(CC(=O)N1CC(CN=[N+]=[N-])C1)(C1CC1)NC(C(=O)NC(C)C)=O CC(C)(C)CC(=O)NCC1(C(C)(C)C)CCN(C(=O)COCCCF)C1 N#Cc1ccc(-n2cncc2NC(=O)C(O)CF)cc1 C1(C)(CCC)CCCN(C(=O)CC2(C)CCN(C(c3cnnn3CC)=O)C2)C1 N1(C(CC2(OCC)CC2)=O)CCN(C(=O)CCOC(C)=O)CC(O)C1 O=C(CCCCC1CC1)NCC(O)CCNC(=O)C(c1ccccc1)O C(CCCCC(=O)NC1CCCC(NC(c2ccc(F)cc2Cl)=O)C1)OCC N1(C(c2c(CCC)nsc2N)=O)CC2(CC)CC1(CNC(=O)C(O)C1CCC1)C2 C1(NC(CSCC=C)=O)CC(F)CN(C(c2ccc(O)c(CO)c2)=O)C1 Cc1ccc(Cl)cc1C(=O)NC(C1CCCN1C(c1cc(C(C)(C)C)no1)=O)C c1(C(C(=O)NCCC(Cn2cc(C3(C)CCCO3)nn2)F)O)ccc(F)c(Br)c1 N1(C(=O)CC2CC2)CC(Cc2ccc(F)cc2)CC1Cn1cc(C2(O)CC2)nn1 C12(C(=O)NCCC(C)NC(c3csc(C4CCCCC4)c3)=O)CCCC1C2(F)F CCC(C)(C(=O)NC(C1(O)CN(C(c2cc(CN(C)C)on2)=O)C1)C)OC CC1CN(C(C2CCCN2C=O)=O)CCN(C(=O)C(O)CC2CCCC2)C1 Cc1cc2[nH]c(C(N3CCN(C(C4CC=CCC4)=O)CC3C)=O)cc2o1 c1(C(N2CC(C(N3C(C(N)=O)CCCC3)=O)C2)=O)cccc2ncc(Br)cc12 Cc1scc(C(=O)NCCC2(O)CN(C(c3ccncc3O)=O)C2)c1C c1(C(=O)OC)cccc(C(=O)NC(C)CNC(C2CCCC(O)C2)=O)n1 CCCCCCC(C)(C)C(=O)N(CC(C)(C)CNC(C1CC12CCCOC2)=O)C CCC(CC(=O)NCC1CCC1C(=O)NCC(C)C(F)F)C1CCC1 N1(CC(=C)Br)CCc2ccccc2C1CNC(c1c(C)cc(F)cc1C)=O c1(C(=O)NC(CC(C)NC(C(C=C)c2ccccc2)=O)C)cc(CC)cnc1O N1(C(CCc2ccc(C)s2)=O)CCC(C)(C)C(NC(C2(C)CCCCC2)=O)C1 C12(NC(CN3CC(C)(C)C3)=O)CCN(C(C3(C#N)CC=CC3)=O)CC1C2 c1(OCCC)ccc(C(=O)NCCC(C)N(C)C(c2cc(Cl)no2)=O)cc1OC c1(OC)c(F)cc(C(=O)NC2CC3(C2)CC(C(=O)Nc2ncc(Br)s2)C3)cc1F C1(C(=O)NCc2cc(OC)ncn2)CC(F)(F)CN1C(=O)CCc1ccon1 O=C(C1=C(Cl)CCCC1)NC1CC1NC(C1CC1(Cl)Cl)=O N1(CCC)CCN(C(=O)C(C2CCCN(C(=O)CCC(C)N(C)C)C2)C)CC1 N1(C(CCOCCOCC)=O)CCC(C(=O)NC(CO)(CO)CO)C(C)C1 c1(OC)cccc(OC)c1C(=O)NCC(C)(O)CNC(c1occ2c1CCC2)=O c12ccc(cc1)SC2.C1(C(C)(C)NC(CCSC)=O)CCOCC1 c1(CC(N2CCOCC(NC(C#CC(C)C)=O)C2)=O)ccc2c(c1)CCC(=O)N2 c1(NCCNC(=NCC)NCC(n2ccccc2=O)C)ccc(C)cc1C C(=O)(C(C)CCC(C)(C)C)NCC1(CNC(CC(CC)C(C)C)=O)CCCCC1 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CC(NC(=O)C(C)(Cl)Cl)CCC(O)C1 Cc1ncccc1C=CC(=O)NCC1(F)CCCN(C(=O)C(C)CC(N)=O)C1 N1(C(CCS(=O)(=O)NC)=O)CCCC2(CCC(=O)N(c3cccc(C)c3)C2)C1 C1(CNC(=O)COC(F)(F)F)CCCN(C(=O)CCN2CCCC2=O)C1 N1(C(C(C(CC)CC)OC)=O)CCOC2CN(C(=O)CCP(C)(C)=O)CC12 C=Cc1ccc(C(=O)NC2(CNC(=O)Cc3cc(Cl)cs3)CCOCC2)cc1 CC1CN(C(c2cc(CNC(c3ccc(N)cn3)=O)no2)=O)C(C)CO1 C1(C(=O)NCCC(C)(C)NC(C2CC3(CCC3)CO2)=O)CCCCC12CCC2 c1(-c2ccc(CNC(N(CCN(c3ccccn3)C)C)=O)o2)ccccc1Cl c1(C(=O)NC(c2nocc2C(=O)NC2(C)CSC2)C)nc(=N)cc[nH]1 C1(NC(CNC(C=C(C)C(=O)O)=O)C(=O)Nc2cccnc2)CC2(CNC2)C1 N1(C(c2scc(C)c2)=O)CC(NC(c2csc(C(C)(C)C)n2)=O)C2(CCC2)C1 c1(C(=O)NCC2(C)CCN(C(C3C(CC)C3)=O)CC2)cc2c(nn1)CCC2 C12(NC(N3CCCC(NC(CC(C)CF)=O)C3)=O)CC3CC(CC(C3)C1)C2 c1(C(=O)NCC2N(C(C3CCCN(C)C3)=O)CCC2)ccc2c(c1)nnn2C c1(N(C(CCNC(=O)NC2C(OC)CCC2)=O)C2CC2)cncc(Cl)c1C C1(C)(C(N2C(C)(C(=O)OC)CC2)=O)CCN(c2cc(C(F)(F)F)ccn2)C1 C1(CC(=O)NC(CC)CN(C(=O)C=CC=C(Cl)Cl)C)CCNC1=O N1(C(C(c2ccco2)NC(CCOC)=O)=O)CCCN(C)CCC1 C1(C(N(CCOC)CCNC(C23COCC2C3)=O)=O)COc2cc(F)ccc2C1 c1(NC(=O)OC)ccccc1NS(=O)(=O)CC.C1(=O)CN1C1CC1 N1(C(=O)OCc2ccccc2F)CC2(CCCN2c2ccncn2)C1 c1(C(N(CC(=O)NC(CC#C)CO)CCOC)=O)ccccc1F Cc1cc(C)c(C(=O)NCC2(C)CCN(C(=O)Cn3cnc(Br)n3)C2)cn1 c1(NC(=O)NC(c2cccc(OC)c2)Cc2ccccc2Cl)cc(F)ccc1Br C1(C(C)NC(c2n(CC)ncn2)=O)CCN(c2ncncc2I)CC1 S(=O)(=O)(c1ccc2c(c1)CCN2C(=O)Nc1ccccc1)Nc1scc(NC)n1 N1(C(C#CC(=O)N(C)C)=O)CCC(C2CCN(C(C3CC4(C3)CC(F)C4)=O)C2)C1 c1(C(=O)NCc2nc(CNC(c3c(CC)occ3)=O)sc2)[nH]c(C)nc1C c1(C(=O)NC2C(NC(c3nc(CCC)oc3)=O)C2)cncc(-n2cnnn2)c1 C1(C(=O)NC(C(C)(C)C)CNC(C2CC2(F)F)=O)CC2C(C1)C2(F)F N1(C(c2c(CC=C)cccc2)=O)CC2(CNC(C3(C)CCCO3)=O)CC(F)(C1)C2 C(=O)(CCCCCC(C)O)N(CCC)CCNC(=O)C(c1ccc(F)c(F)c1)C C(=O)(CCC(CC)OC)NCC(CCCC)NC(C1CC(C)(F)C1)=O C(C)(C(=O)NCC1CN(C(N)=O)C1)=CC N1(C(Cc2c(C)cccc2)=O)CC(C2CCCN(C(=O)CCN3CCCC3)C2)C1 Cc1sc(Cl)c(C(=O)NC2CCN(C(c3ccc(C(F)(F)CF)cc3)=O)C2)c1C C1(NC(CCCc2nc(C)sc2)=O)CC(C)N(c2nnc(C(C)C)o2)C1 c1(OC)cc(=O)n(C)cc1C(=O)NC(CO)C(C)NC(=O)C(C)N1CCC1 C1(OCC)CCC(CN=C(NC2CCCC2)NC2CC=CCC2)CC1.C1CO1 c1(C(N2CC(CNC(CCC)=O)CC(C)(C)C2)=O)cc2c(C)cccn2n1 C1(NC(CCN(CCCCC)CC)=O)(CO)CCN(C(=O)C=Cc2cnc[nH]2)C1 C1(NC(c2cnc(C)s2)=O)CC2C1CCN2C(=O)CN1CCN(C2CC2)C1=O C(=O)(C(C)CC(C)C)N1CCC(N(C(=O)COCCCOC)CCCC)CC1 c1(NC(C2N(C(c3ccc(C)cc3)=O)CCCC2)=O)ccn2ncc(F)c2c1 C1(NC(=O)C(F)=CC2CC2)CCN(C(c2coc(C3CC3)n2)=O)CC1CO C1(C(=O)NC2(CF)CCN(C(=O)C=CC3CC3)C2)CC2CC1C1C2C1(F)F C1(CC(N2CCC(C)(NC(C3CC(=C4CCC4)C3)=O)C2)=O)CCC2(CCC2)O1 CCCCC(CC)C(=O)NC1CC12CCN(C(=O)C(C)(C)CCC(=O)OC)CC2 S(=O)(=O)(c1cnn(-c2ccccc2)c1F)NC(c1ccc(C(CC)C)cc1)=O c1(CC(N2CC(O)(C(C)NC(=O)C(F)=C3CCCC3)C2)=O)cccc2c1OCC2 CCC(COC)C(=O)NCC(C)(C)C(=O)NC(c1nc(C)cs1)C C1(C)(CNC(C(CCC)N(C)C)=O)CCCN(C(=O)C=COC(=O)OC(C)(C)C)C1 C(C(C)C(=O)NCCCN(C(=O)CSc1nc[nH]n1)CC1CC1)OCC c1(NC2(c3n(CC=CC)nnn3)CCN(C)C2=O)ccc2ncccc2c1 C1(C(=O)NC2CCCN(CC(=O)O)C2=O)CNc2cccc(Br)c2O1 c1(C(=O)NC(C)(CNC(c2cnc(Cl)s2)=O)C2CCC2)ccnc2cc[nH]c12 C(=O)(C(F)C(C)(F)F)N1C(C(=O)NC(C=C)(C)CC)C=CCC1 c1(C(C(N2CCC(C(C)(C)NC(COCC(=O)NC)=O)C2)=O)C)ccccc1F CN1C(=O)OCC1C(N1CCOC(CNC(=O)Cc2cccc(C(F)F)c2)C1)=O Cc1ccc(Cl)c(O)c1C(=O)NC1CCCC1NC(c1nc2ccccc2s1)=O N1(CC)CC(C(=O)N(C(C)CNC(c2c(C)cc[nH]c2=N)=O)C)c2ccccc21 c1(C(N(C(CNC(c2ncoc2-c2ccon2)=O)C2CC2)C)=O)ccccc1 N1(C(CC2N(C(C3C(C)CCC3)=O)CCC2)=O)CCC(CO)CC1 C1(CNC(CSCCCC)=O)CCC(N(C)C(c2cccc(F)c2)=O)CC1 c1(C(=O)NC2C(CNC(=O)CC3CC=CC3)C2)ccn2ncc(Br)c2c1 N1(C(C2CN(C)C(=O)N2)=O)CC(N(C)C(c2ccc(=O)oc2)=O)C2(CC2)C1 C1(CCCNC(=O)CCc2nccs2)CN(C(=O)CCC2CC2(Cl)Cl)CCO1 Nc1cccnc1C(=O)NC(c1ccccc1)C(N1CC=CC(O)C1)=O S(=O)(=O)(c1ccc2c(c1)CCCC2)N1CCC(O)(CNC(C2(CN)CC2)=O)CC1 N1(C(c2cc(OC)n[nH]2)=O)CCN(C(c2ccsn2)=O)C(c2ccccn2)C1 C(=O)(CCCCC(C)CC)NC1(CC=C)CCCN(C(c2cc(CO)[nH]n2)=O)C1 C1(C(N(CCCn2cnnc2)C)=O)CCC2CCC1N2C(=O)OC(C)(C)C C1(CNC(c2cc(OC)ncc2Cl)=O)CN(C(c2cocn2)=O)CC2(CCC2)O1 Cc1cccc(C)c1CC(N1CCC(NC(=O)CC2CCC(=O)C2)CC1C)=O C(=O)(N=c1ncn(C2CCS(=O)(=O)C2)[nH]1)C1C(C)CCCC1 C1(OC(C)(C)C)CN(C(=NCC(C)(C)c2ccc(C)s2)NC2CC2)CCO1 N1(C(c2c(NCC)nccc2)=O)CC2CC(C)N(C(=O)CCOC3CC3)C2C1 C1(C2CC2)(CNC(c2cc(C)ncc2C)=O)CCN(C(C2(C)CCSCC2)=O)C1 N1(C(C(C)C)=O)CCCCC2(CCN(C(c3cccc(C4CC4)n3)=O)C2)C1 CC1(C)CC(NC(=O)C(C2CC2)NC(=O)CC2C(C)(C)C2(C)C)CO1 C1(NC(c2ccccc2F)=O)CN(C(=O)NC2CCC2)CC1c1ccccc1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C2N(C)C(=O)CC2)=O)C(F)C1 C(=O)(C1CCCc2ncnn21)NC1C(NC(C2CCN(CC)CC2)=O)C=CCC1 N1(C(c2c(C)nc(CNC(CC(CC)C(C)C)=O)o2)=O)CCC2(CNC(=O)O2)C1 C(=O)(CN=c1cc[nH]cc1)N1CCCC(C(=O)Nc2c(C)noc2C)C1 c1(C(=O)NC(C2N(C(c3ccc(C(C)C)[nH]3)=O)CCC2)C)cc2c(ncn2C)[nH]1 C1(CCNC(CCCC#C)=O)CC2CCC(C1)N2C(c1c(CC)noc1C)=O n1(CC)cc(C(N2C(CNC(C3(C)CSC3)=O)CC2)=O)c(C2CC2)n1 C1(CC(=O)NC2CCCC(C(C)C)C2)CC2(C1)CN(C(=O)Nc1ccccc1)C2 C1(C)(C(=O)NC(CCCNC(c2c(C)nn(C)n2)=O)(C)C)CCCCCC1 C1(NC(CCN(C)CC)=O)(CNC(c2cncc(Cl)n2)=O)CCCCC1C C(CCCCCNC(C1CC1(F)Cl)=O)NC(C1(CC=C)CC1)=O Cc1cc(-c2cn(C3(C(N4CCC(CC5CCOC5)C4)=O)CC3)nn2)cc(C)c1 N1(C(C2(C)CCCO2)=O)CCC(C2CCN(C(c3c(F)ccnc3F)=O)CC2)C1 CC(C(C)C(=O)NCCC1(C)CCOCC1)NC(c1ccn(C)c1)=O C1(NC(C(F)OC)=O)CCN(C(=O)CCCS(N)(=O)=O)CCC1CO c1(OC)cccc(C(=O)NCCN2C(=O)C3CC3C2)c1OC.N(C)(C)C(C)C N1(C(c2ccc(CC)s2)=O)CC(NC(=O)C(C2CC2)SC)CC2(CCOCC2)C1 C1(NC(CCC(=C)Cl)=O)CCSC12CN(C(c1nc(C)c(C)[nH]1)=O)C2 CS(=O)(=O)c1cc(C(N2CCCC23CN(C(c2csc(Br)c2)=O)C3)=O)ccc1F N1(C(C2CCC(C)CC2)=O)CC2CCN(C(=O)CCC(CF)CF)CC12 c1(N(C)Cc2ccc(C(=O)OCC)c(OC(F)F)c2)cccc(F)c1C#N CN1CCC(C(F)(F)F)(CN(C(=O)C=CCN2CCC2)C2CC2)C1.C1(=O)CCN1 C(=O)(C1=C(NC)CC1)NC1C(CNC(c2c(CC)nc[nH]2)=O)CCC1 N1(C(CCN(C)C)=O)CCC(F)(C(=O)NC2CC(C)(N(C)C)C2)C1 CCCC(C(=O)NCCCC(C)NC(c1ccc(OC)o1)=O)OCC c1(C(N2CCC(OC)(CNC(=O)CC(C)SC)C2)=O)n[nH]c2c1CCOC2 c1(C2C(C(N(CCN(C(c3cnnc(O)c3)=O)CC)CC)=O)C2)ccc(O)cc1 C1(CNC(c2cc(C)nc(C)c2)=O)CC2CCC1N(C(=O)COc1ccsn1)C2 C1(CCNC(C2CS(=O)C2)=O)CCCN(C(=O)CSc2n[nH]c(O)n2)C1 N1(C(c2n(CC)nnc2)=O)CCC(NC(c2ccsc2C)=O)CC1C N1(C(CCOCC(C)C)=O)CCCC(NC(=O)CN(C)CCOC)C1C N1(C(C2C(OC)C2)=O)CCCC2(CCN(C(C3CC4(CCOCC4)C3)=O)CC2)C1 C1(C(N(CCNC(c2c(C)ccc(OC)c2)=O)C)=O)CCCC12OCCO2 C1(NC(=O)CC2CC(CF)C2)CC(F)CN(C(=O)CCc2cccnc2)C1 c1(OC)cc(N(C2CC3CNCC3C2)C(C2=CC=C(F)SN2)=O)nc(OC)n1 C1(C(N(C)CC2(OC)CC2)=O)CSCN1C(c1ccns1)=O Cc1cn2c(n1)CCC(C(=O)NCC(C)(C)NC(c1ccc3cc[nH]c3n1)=O)C2 c1(N2CC(C(C)NC(=O)COCc3ccccn3)C2)ncnc2[nH]ccc12 Cc1cnsc1C(N1CC(O)(C(C)NC(c2ccccn2)=O)C1)=O C(=O)(C1=CCC(NC(=O)CC2C(=O)NN=C2C)C1)N(CCCOC)C c1(C(N(CC(C)N(C)C(c2n[nH]c(C3CC3)n2)=O)C)=O)cc2c(nc1O)CCC2 CC(CC(=O)N1CC2(CC(NC(=O)CN3CCSCC3)CO2)C1)P(C)(C)=O N1(C(C2N(C(C(CC=CC)C)=O)CC(=O)C2)=O)CCN(C)CC(O)C1 Cc1c(C(N2CC3CC(NC(C4CC4C(N)=O)=O)C2C3)=O)[nH]c2c1C(=O)CCC2 c1(C(N2C(C(N(C(=O)N)CC)=O)CSC2)=O)nnn(C)c1C.C(C)C1CC1 c1(C(=O)NC(CNC(C(C=C=C)C)=O)(C)C2CC2)ccc(O)c(OCC)c1 N1(C(C=C(CC)C)=O)CC2COCCC2(NC(=O)CSc2cccc[n+]2[O-])C1 n1(CCCOC(=O)NC(Cc2cc(C)no2)=O)nnc2ccccc12 C1(CN(C(=O)CCC(=O)N2CCCC2)CC)CCCN(C(c2ccncc2)=O)C1 C1(C(N2CCC(CNC(CSC(C)C)=O)C2)=O)CC2CSCC(C1)C2(F)F CCC(C)CC(=O)C(=O)N1CC=CC1Cn1cc(-c2cccc(C)n2)nn1 C1(C(=O)NCCCC(C)NC(=O)C(C2CCCCC2)C)(OCC)CCCCCC1 C1(C#N)(C(N2CCC(CCNC(C=C(CCC)CCC)=O)C2)=O)CC2CC2C1 N1(C(CS(CC)=O)=O)CC2CC(O)C1C2NC(=O)CC1CSC1 N1(C(CCCOCC)=O)CC2CC(C(N3CCNC(=O)C3CCO)=O)CC2C1 c1(C(=O)NC2C(NC(C(C(C)(C)O)F)=O)CC2)cc2c(cc1O)OCO2 N1(C(CC(C)(C)N(C(=O)CCCn2cccn2)C)=O)CCC(C2CC2)CC1 C1(=CC(=O)N(C2CN(C(C3CCC4(CC4)C3)=O)CCC2O)C)CN2CCC1CC2 c1(C(N2CCC(C(C)NC(c3ccc(Br)o3)=O)C2)=O)cnc2c(c1)OCCN2 N1(C(C2CC2c2cccc(Br)c2)=O)CC2CCN(c3ncccn3)C2C1 N1(C(c2cc(C)ns2)=O)CC2CCN(C(=O)CC(C)F)C2C1 CCCC(CC)CCC(=O)N1CC(NC(c2ccc(OC)c(Cl)c2)=O)C(SC)C1 C1(C)(C(=O)NC(C(N2CC(O)(C(=O)OC)C2)=O)C)CCC(C)C1 N1(C(C2CCN(C(c3cc(SC)oc3)=O)CC2)=O)CC(F)(F)CC1CN(C)C CN=c1nc(C(N2CCC3(NC(=O)CC4(CSC)CC4)CC3C2)=O)cc(C)[nH]1 Cc1ccc(C(N2CCCC2C(N2CCC(C)CC2)=O)=O)c([N+](=O)[O-])c1 c1(CNC2CC3(CC(NC(Cc4cccc(C)c4)=O)C3)C2)c(Cl)cc(F)cc1Cl c1(C(C(=O)NCCCF)N(CC2CCCCC2)CC2CC2)nc(Cl)ccc1Br C(=O)(C#CC1CCCCO1)N1C(COC)CN(C(=O)Cn2ccnn2)CC1 c1(NC(C(CSC)(C)NC(=O)CC2CCCC3CC23)=O)cc(O)ccc1F C1(NC(c2cccc(NCC)n2)c2nnnn2C(C)C)CC2(CCOCC2)C1 Cc1ccc(C(N2CCC(=CCNC(c3c(C)nc(C)n3O)=O)CC2)=O)nc1C N1(C(=O)NC2C(CCC)CCC2)CCS(=O)(=O)C(C)(C)C1 c1(OCC(=O)NCC2CCN2C(=O)CC2CC2)ccc(Br)nc1 C(=O)(CC(C)C(F)(F)F)NC1CCCN(Cc2nc(C)oc2)C1 C=CCN=C(NCc1ccc(-c2ccccc2)cc1)N1CCN(CC)CC1.C1CC1 N1(S(CC=C)(=O)=O)CC2OCCN(c3ccn4ncc(I)c4n3)C2C1 C=CCCCC(C(=O)NCc1[nH]nnc1C)NC(C1=NOC(C)C1)=O C1(N(C(c2cnn(CCCC)c2C2CC2)=O)C)CCCCN(C(C2CSC2)=O)C1 c1(NC(=O)CC2(NCC3CCOCC3)CCC2)cc2c(Br)cccc2s1 C(CCS(=O)(=O)c1ccc(Cl)cc1)C(=O)NCc1cnc(C(C)C)[nH]1 c1(OC)cc(N)c(F)cc1C(=O)NC1(CNC(c2cncnc2C)=O)CCC1 C1(C(N(C(CNC(c2c(SCC)cccc2)=O)C)C)=O)CCc2n[nH]cc2C1 CC(N=c1[nH]c(=N)[nH]c(=NCCCOCC(F)(F)F)[nH]1)c1ccccn1 N1(C(CC)=O)CC(CNC(C2C=CCC2)=O)C(F)(F)C1 Cn1c(C(N2CCC(O)(Cn3cc(C4CCC4)nn3)C2)=O)cnc1S Cc1ccc(O)c(C(N2CC(O)CC2(C)C(=O)NOCC(N)=O)=O)c1 CC1CCCC1(C)NC(c1conc1CNC(C1CCCN1C1CC1)=O)=O c1(OC)c(C(=O)NC(C2(O)CN(C(C3CC4COCC4C3)=O)C2)C)cccc1C N1(C(c2c(C)cnnc2)=O)CCC(O)(CNC(C2(C#N)CCOC2)=O)CC1 c1(COC)csc(CNC(C2CCN2C(=O)CNC(=O)C(C)(C)C)=O)n1 N1(C(Cc2c(C)n[nH]c2)=O)CC2(NC(C3CCS(=O)(=O)C(C)C3)=O)CCC1CC2 C(=O)(CCC(O)C(C)(C)C)NCCCCC(C)NC(c1c[nH]nc1C(C)(C)C)=O c1(CC(=O)N(CC(C)C)CC(C)C)csc2ccc(Cl)cc12.c12cccc(c1)N2 CC1(O)CCC(C(=O)N(C2CCC2C(N2CC(C)(CO)C2)=O)CCO)CC1 C1(C(N2CCCC(C(=O)NCC3(C4CC4)CCC3)C2)=O)CCOC(=O)CC1 N1(CC(=O)NC2CC(CNC(C3CCCCCC3)=O)CC2O)C(=O)CCCC1=O N#Cc1cc(CNCC2CC(c3cccc(F)c3)(F)C2)cc([N+](=O)[O-])c1 CS(=O)(=O)C1CCCC1C(N1CC2(CC(NC(=O)C3=NOCC3)CO2)C1)=O N#CC1(CN2CCC2C2CC2)CC2CC2C1 C1(C(N2C(C(C)C)CC2)=O)CN(C(=O)CC2CC(=O)C2)CCN1C c1(-n2c(CN3CCCC3)ncc2)ccc(Nc2ccc(SC)cn2)c([N+](=O)[O-])c1 c1(C(=O)NCCN(c2nccnc2F)CCC)ccnc(CO)c1 c1(OC)cc(C(=O)NC2CCC(C)(CNC(C3(N=[N+]=[N-])CC3)=O)C2)cnc1O C(CCCC(=O)N1CCC(O)(CNC(c2cocc2C)=O)C1)(OC)OC C(=O)(C(F)(F)C(O)C(C)C)N1CC(O)(CCNC(C(CC=C)CC)=O)C1 c1(OC)ccc(CN2CCCC2(C)C(=O)NC(C)C(=O)N(C)C2CC2)c(OC)c1Cl O=C(CCCC1CCC1)NC1CC(CNC(C2CC=CCO2)=O)C1 C1(CC)CN(c2nnnn2CCOCc2ccccc2)CC1OC CC(C)C(CO)C(=O)N1CCC(C(C)NC(=O)C(C)N(C)C)C1 N1(C(C(C)(C)C2CCCCO2)=O)CCOC2(C1)CN(C(C1CC(=C3CC3)C1)=O)C2 CC(CCc1cn[nH]c1)N=c1[nH]c(=NC2CCC2)[nH]c2c1CSC2 N1(C(C2(F)CC(C(N)=O)C2)=O)CC(O)CC1CNC(=O)C(F)=CCCF c1(C(=O)NCC2CC3CN(C(C=CCCC)=O)CC32)cc2ccsc2c(O)n1 c1(CC)c(C(=O)NC(C2CCCN(C(c3cn(C)[nH]c3=N)=O)C2)C)csc1C O=C(CC1CCOc2ccccc21)NC1CN(C(=O)C#CC2CC2)CC12CC2 C(=O)(CCCCC(=O)N1CCC2CN(C(=O)CCCC(C)=O)C2C1)OC Cc1nnc(C(N2CCCC2c2cccs2)C(=O)NCC(C)C)n1C c1(CCc2c(F)cccc2)nccc(=NCc2csc(CCC3CCCS3)n2)[nH]1 N12CC3CC1C3NCC2.CC1CC(C)(CC2(C3=CC=C3c3cnc(O)s3)CC2)C1 Cc1[nH]c2ccc(Cl)cc2c1C(=O)NCC1C2CN(C(C3CCSC3)=O)CC12 CCC(COC)C(=O)NCC(C)CC(=O)N1CCCC1C(=O)N(C)C c1(C(=O)NC2(CCC(=O)NCCOCC(=O)NC)CCCC2)nnc(O)nc1O C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NCCNC(C1(C)N(C)CC(O)C1)=O C1(CNC(c2n(CC)ncn2)=O)CC12CCN(C(=O)CC1CCCOCC1)CC2 CC#CCCCCNC(=O)CCC(C)NC(c1cc(OC)nn1C)=O Cc1cccc2c1CC(C(=O)NC1CC1NC(=O)Cc1ccc(F)cc1F)O2 C1(CC(=O)NCC2CCC(F)C2)CCC(F)(F)C1.C12(CCCC1)C(=O)NC2 c1(OC)cc(C)ccc1C(N1CCCC(O)(CNC(=O)CNN2CCCC2)C1)=O C1(CN(C(CCc2onc(CC)n2)=O)C)CCN(C(C2CC(C)C2)=O)CC1 C(=O)(N1OC2CCC1CC2)C1CCCN(C(COC2N(C)CCC2)=O)CC1 c1(C(N(CCN(C(=O)CN2CCC(C)(O)C2)CC)CC)=O)ccc2nc(O)oc2c1 C1(C(=O)Nc2c(C)ncnc2)CCCCN(C(=O)CCCC2CCCO2)C1 C1(CNC(C2(SC)CC(O)C2)=O)C2CCC(C2)N1C(=O)C=CC(C)(C)C CC1(C)CC(C(=O)NCC(C2CCCC2)NC(c2cccnc2)=O)C1 c1(C(N(C2C(C)CCN(C(C(C)OC(C)C)=O)C2)C)=O)cnn2ccccc12 C1(C(N(C(CNC(CNC(C)=O)=O)C2CC2)C)=O)C=C(C)CS1 c1(C(N(C2CCCCN(C(c3c(C)coc3C)=O)C2)C)=O)nc(Cl)c(=O)[nH]c1N c1(CC)cc(C)nc(N(CCCNC(C2CCC(C)C(C)C2)=O)C(C)C)n1 N1(C(C(N)=O)=O)CCCC(n2cc(-c3csc(C4CC4)n3)nn2)C1 N1(C(C(=O)NCCS(C(C)(C)C)=O)=O)CCOC2(COC(C)(C)C2)C1 c1(SC)cc(C(N2CCC(NC(c3cc(=O)n(C)cn3)=O)C(F)C2)=O)ccc1F c1(OC)cc(C)c(NC(C2CCN(C(C3CCC3OC)=O)C2C(C)C)=O)cn1 Cc1nc(CNC(c2ccccc2OC(F)F)=O)nc(NNC(=O)N(C)C)c1C N1(C(C2CN(C)C2)=O)CCC(NC(=O)CCC(C)(C)O)C12CCCC2 Cc1n[nH]c(C)c1CC(=O)NC1CCC(NC(=O)CCN2CCCCC2C)C1 c1(NC(C2CCN(Cc3ncco3)CC2O)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(C(C)C2CC2)=O)CCC(O)C2(CCN(C(=O)CCCNC(=N)N)CC2)C1 C1(OCCC)(CNC(=NCC2CC2)NC2CSC(C(C)C)C2)CCCCC1 C1(F)(CNC(c2c(CCC)cccc2)=O)CCCN(C(=O)C(C)(C)Br)C1 C(=O)(C1CCCn2cc(C)nc21)C1OCC(=O)N(CC)C1c1nnc(COC)o1 N1(C(CCOC(C)=O)=O)CCC2CCN(C(=O)CCc3nncn3C)CC2C1 C1(C(=O)NCC2C3CN(C(c4n(C)ncc4)=O)C2C3)Cc2ccccc2N1 Cc1nn(CC(=O)NC(C)(CNC(C2(CCF)CCC2)=O)CO)cc1Br C1(C(C(=O)OCC2CN(CC3CC3)C2)NC(C2CC2(Cl)Cl)=O)CCCCC1 Cc1nc(C)n(CC(=O)NCC2CSCN2C(=O)C(c2ccn(C)n2)C)n1 c1(C(C#N)NC2C(NC(C(C)=C3CCCC3)=O)C2)ccccc1 C(c1cccnc1C)=CC(N1CCCC(CNC(c2c(C)coc2)=O)C1)=O N1(C(c2nc(COC)oc2)=O)CC2CC1CN(C(c1cnc3ccnn3c1)=O)C2 N1(C(COCCOCCOC)=O)CC(NC(c2snc(Cl)c2Cl)=O)C(O)C1 C1(NC(C2N(CC(C)C)CCC2)=O)CN(C(=O)CCOCC2CC2)CC2(CC2)C1 c1(CC(=O)NC(C(C)NC(CCC#C)=O)C)ccc(Br)cc1C#N C1(C(=O)NC2(C(=O)O)CCC(OC(C)(C)C)C2)CCc2cncn2C1=O Cc1ccc(-n2cccn2)cc1NC(=O)CNCC(F)(F)F N1(C(CC=CCC)=O)CCC(F)(F)C(CNC(C2Cc3nnc(C)n3C2)=O)C1 c1(C(=O)NCCON)nc(Cl)cs1.c12n[nH]cc1C(=O)N(C)C2C CC1CN(C(=O)CC2CCCCC2C)CCC1CNC(=O)C(=O)N(C)C c1(OCC)c(C(=O)NCC(C)CNC(c2cnc(OC)c(C)c2)=O)cccc1F C1(CNC(C2CN(C(C)C)C2)=O)CCCCC1O.C1(=O)C(O)C2CN1C2 CN1CCN(C(C2(C#N)CC(=O)C2)=O)CC1C(N1CC2CC2C2CC12)=O c1(C(N2CC3C(NC(C(C)O)=O)(CC3)C2)=O)cccc(S(=O)(=O)CC(F)(F)F)c1 CCCC(C(=O)NC1CC12CCN(C(=O)C(O)C1CCCC1)C2)C(C)C N1(C(CCCC=C)=O)CCC2CCC(C1)N2C(c1cc(C)c(CC)nc1O)=O CN1CCCC(O)(CC(=O)NCCC2CC(NC(C3(C)SCCCS3)=O)C2)C1 C(=O)(CCC(=O)NC1C2CCN(CCCc3csc(C4CCC4)n3)C12)NC.NC C1(C(C)C)N(C(c2ccc(CNC(C3COC(=O)N3C)=O)nc2)=O)CC1(C)C CCCCC(C)CCC(=O)N1CC(C(N2CC3CCC(C2)O3)=O)CC(F)C1 N1(C(C(CCC)C)=O)CCC2(CCCN(C(c3cncc4[nH]ccc34)=O)C2)C1 N1(C(CC(=O)OC)=O)C(C)C(C(=O)NCC(C)(O)C2CCCC2)C1C N1(C(C2N(C)C(=O)CC2)=O)CC2=C(C1)CN(C(=O)Cc1cccc(Br)c1)C2 C12(NC(c3cocn3)=O)CCCC1N(C(c1cnc3ccnn3c1)=O)CCC2 c1(C(=O)NC2C(C(N(CCN(C(=O)OC)C)C)=O)CC2)cccc2nccn12 Cc1cc(Cl)cc(C)c1C(=O)N(CCCCCNC(c1cccc(F)c1O)=O)C c1(OC)ccc(CC(C)(C)C(=O)NCC2CCN2C(c2cnn(C)c2)=O)cc1OC C1(CC(=O)NCC(=C)CCNC(=O)C(C)(C)C2CCCC2)CCCOCC1 CC1CN(C(C2C3CCCOC23)=O)CC(C(=O)NC(C)C(C)(C)C#N)O1 C(=O)(CCC(=O)NCC1CCCC1NC(c1ccc(C2COC2)cc1)=O)NC Cc1cc(F)ccc1C(N1CCOC(c2ccccc2Cc2ccccc2)C1)=O C(CC)(C(=O)NC(CNC(=O)C(C1CCCC1)OC)C(C)C)OCCOC c1(SCCNC(=O)CCc2cncnc2)ccc([N+](=O)[O-])cc1 N1(C(C2CCN(C)C2=O)=O)CCC(C)(C(=O)Nc2ccc(CO)c(F)c2)CC1 C(=O)(C=C1SCC(=O)N1C)N1C2CC(NC(COC)=O)C1CC2 CC(C(C)C(=O)NC1CC1O)NC(=O)Cc1cc[nH]c1 CC1C=C(C(=O)NCC2CN(CC(=O)OC(C)(C)C)CCN2C)CC1 c1(C2(C(=O)NC(C)C(C)(C)N)CC2)ccc(Cl)nc1.C(=O)(CC(=O)N(C)C)NCC c1(C(=O)NC(CC2CN(C(C(CC=CCC)C)=O)C2)C)cc(=O)c(OC)cn1C c1(C(C(=O)NCC2(CNC(CCOCC#C)=O)CC2)F)cccc(F)c1 C1(N(C(c2cnc(C)nc2C(C)C)=O)C)CC2CCC(C1)N2C(c1cnsc1)=O C(=O)(C(O)C1=CCCCC1)NC1(CC)CCN(C(c2nccc(C#C)c2)=O)C1 CC1(C)CC(C(=O)NCCc2cccnc2)CN1C(=O)Cc1cn[nH]c1 C1(C(=O)OC)N(C(c2ccc(CNC(C3CC3C(=O)OC)=O)cn2)=O)CC1(C)C C1(C(=O)NC2CC(CF)C2)CC12C1CC3CC(C1)CC2C3.C1(NC(=O)CO)CCC1 C(=O)(C(C)(F)C(=O)NC1CC(CNC(=O)CCCc2cc(C)no2)C1)OC CCCCC(O)C(C)C(=O)N1C2CCCC1CN(C(c1nn(C)cc1C)=O)C2 c1(NCCNC(C)=O)nccc2cc(C)ccc12 c1(CC)ccc(N)c(C(=O)NC(C)CN(C)C(c2ccc(OC)c(OC)c2)=O)c1 C(=O)(C1=Cc2ccccc2C1O)NCC1CCCN(C(CNS(C)(=O)=O)=O)C1 C1(C)(C(=O)NC2(CNC(C(C(=O)OC)C)=O)CCC2)CCN(C)C1=O C(CCN=C(NCC(c1ccc(OC(F)F)cc1)C)N1CCSC(C)(C)C1)OCC C1(C(C)C)C(C(=O)NCCC2CCCC3CC23)CCN1C(c1ccc(O)cc1)=O C1(C(=O)OC)CCN(S(=O)(=O)NC(c2ccc(Cl)cc2)C2CCOCC2)CC1 N1(C(c2ccoc2C2CC2)C(=O)NCCC)CCOC(c2ccco2)C1 C1(C(=O)NCc2oc(C(=O)NC(C3CCCO3)CC)c(C)n2)CC(=O)NC1(C)C CC1CCCCC1CC(=O)NC1CC(CNC(c2c[nH]nc2C(F)F)=O)C1 c1(OC(CN(C(=O)COCC(=O)OC)CC2CC2)C)cc(C(F)(F)F)ncc1Cl.CO C1(C(=O)NC2(CNC(=O)CCC3CCCO3)CCC2)CCCC1F c1(CCNC(=O)CN2CCC(n3cccc3)C2)cn(Cc2ccno2)nn1 Cc1cnc(F)c(C(N2CCCC(n3cc(C(C(C)C)NC(C)C)nn3)C2)=O)c1 Cc1cc(CCNC(C)CCCN(C)C)n(-c2ccccc2)n1 CCCCCCCCC(C1CCCC1C)=O.C12(O)CN(C1)C(=O)NCC2(C)C C1(C(N(c2ccncc2)C)=O)CN(C(C2CCC3(CC2)CC3)=O)CC12CC2 C1(C(N2C(COC)CC2)=O)CNC(=O)CN1C(c1cc(C)oc1C)=O C#CCC(CC(=O)NCCS(N)(=O)=O)NC(c1cncc(Cl)c1)=O c1(-c2ccc(C(=O)OC(C)C)nc2)cc(C(=O)NCc2ccccc2)ccc1F c1(C(n2cc(COc3ccc(Br)c(O)c3)nn2)C)cc2c(cnn2C)nc1O N1(C(C2CC(=C)C2)=O)CCC(C(N2CCC(C(N)=O)C2)=O)C1 c1(C(N2C(C(C)C)C(NC(=O)CS(C)(=O)=O)CC2)=O)cnc(O)c(F)c1 n1(CC)ncc2c(C(=O)NC(c3ccc(C(C)C)cc3)C)cc(C3CC3)nc12 C(CCC(N)C(=O)N1CCC(c2ncc(Br)cn2)CC1)N(C)C N1(c2nccc(OC)n2)CCC2(CCN(C(c3ccc(CO)cc3)=O)CC2)CC1 C1(C(=O)NCc2c(C(=O)Nc3cnc(SC)nc3)con2)OCC2CCCC12 N(C1CCCn2ccnc21)C(C1(C(C)C)CCN(C(=O)C=CCN2CCC2)C1)=O C1(CCN(C(=O)CC2CC3(CCC3)C2)C)CCN(C(c2cscn2)=O)CC1 C12(NC(c3cnc(C(C)C)[nH]3)=O)CC1CN(C(=O)Cc1ccccc1F)C2 c1(OCC)cccc(C(=O)N(C2CCC(NC(=O)CC3CCC3)C2)C)c1 Cc1ccc(COCC(N2CCCC(CCNC(C3CCSC3)=O)C2)=O)cc1 CC1CC(CO)CN1C(=O)CCCCNC(=O)Cc1ccnc(O)c1 Cc1nc(C(=O)NCc2csc(C(=O)N(C)CCOC(C)C)c2)n[nH]1 c1(C(N2CC3C(NC(c4ncc(C)cc4C)=O)(C3)C2)=O)coc2c1CCCC2 N1(c2cc(CCC)nc(C)n2)C2CCC1CC(NC(c1cn(C)cn1)=O)C2 c1(COC)cncc(C(=O)N(C2CC2)CC2CCCN2C(=O)C(F)F)c1 C(C1CN(C(=O)CC2CCCC(C)(C)C2)CC1C(=O)N(CC(F)F)C1CC1)=CC C(C(C(=O)N(CC(=O)NC(C)(C)C)C)C(C)C)NC(c1cc(C)nnc1)=O C#CCC(CC(=O)NC1CN(C(C2CCCC2F)=O)CC1C)c1ccccc1 N1(C(Cc2nc(COC)sc2)=O)CCC(NC(C2CC(=O)NC2(C)C)=O)C(C)C1 C(=O)(CCCCCSC)N(CCN(C(c1cncc(OC)c1)=O)C)C c1(NCC)cncc(C(=O)NCCCCC(C)NC(C2(C)CC3CC3C2)=O)c1 c1(CCNCC(CO)NC(=O)CN2CCC2C2CCCC2)nnnn1C1CCCC1 CC(C)CC(C(=O)NC1(C(=O)N(C)CC2CCCCO2)CCSC1)n1ccnc1 N1(C(C2N(CC)CCOC2)=O)CCN(C(c2cc(C)c(O)nn2)=O)C2CCC12 c1(C(=O)NC2CCC(CNC(=O)C=CC3CCCC3)CC2)ccc2c(c1)OCO2 c1(N2CC2=O)nccc(C2CCCCC2)n1.Cc1cncn1CC(=O)O C1(C(=O)NCc2nncn2C2CC2)CCCCN1C(=O)CCC=CBr C1(CNC(CC(CC)O)=O)CCCC2(CN(C(c3c[nH]c4ncccc34)=O)C2)O1 C1(C(=O)NCC(CN(C(C2(CC)COC2)=O)C)C)CC(c2ccccc2C)=NO1 C1(NC(Cc2c(C)noc2Cl)=O)CN(C(=O)CC2NC(=O)CNC2=O)C(C)(C)C1 N1(CC(=O)N(C2CCCN(C(c3cc(C)c(C)[nH]3)=O)C2)C)CCCNS1(=O)=O c1(C(=O)NCC2C(CNC(c3nn(C)c(CC4CC4)c3)=O)C2)ccc(N)c(N)n1 C1(C2CC2)(CNC2(Cc3ccccc3)CCCCO2)CC2CCCC12 C1(C)(C(=O)NCC2CC(C)N(C(=O)Cc3ccccn3)C2)COC(=O)OC1 c1(C(CN2C(C)CC(N3CCOCC3)C2)C)ccc(Br)c(Cl)c1 C(=O)(CCCCC(=O)N(CC(O)CNC(=O)Cc1cccc(OC)c1Cl)C)OC C1(C(N(CCC(C)NC(c2c(F)ccc(C)c2)=O)C)=O)CC2(CCOCC2)CO1 Cc1sc(Br)c(C(=O)NCC2(F)CN(C(C3CCCC3O)=O)C2)c1C C1(C)(CC)CC(NC(=O)COCC(F)(F)F)CN1C(c1cccc(F)c1OC)=O CCC(C)C(=O)C(=O)N1CC(N(C)C(C2CC(C3CC3)=NO2)=O)C2(CC2)C1 N1(C(CCC(CC)OC)=O)CCCN(C(=O)Cc2ccnc(OC)c2)C(C)C1 C#Cc1ccc(C(=O)NCc2cc(C)c(C(=O)NC(C3CCCCC3)C)o2)nc1 N1(C(c2c(C)noc2)=O)CCCC(NC(=O)CNC(N2CCCC2)=O)C(F)C1 c1(OC)cncc(-c2ccc(NC(=O)CN3CCC(CO)CC3)cn2)c1 Cc1nc(Cl)ccc1CC(N1CCN(C(c2csc(O)n2)=O)C(CC2CC2)C1)=O C1(C(=O)NCC2(F)CC(NC(COC(C)C)=O)C2)CCCN(C)C1 c1(C(N2CC(CNC(C(C)CN(C)C)=O)OCCC2)=O)cc2ccnc(Cl)c2[nH]1 Cc1ccc(C(N2CCC(CF)(NC(=O)CC3CCCOCC3)C2)=O)c(O)c1 c1(C(=O)NC2C(CNC(=O)CN3CCOC3=O)COC2)ccc2cnccc2n1 c1(CCC(=O)C(=O)NCCC(=O)OC(C)C)ccc(Br)cc1.NCC c1(C(=O)NCC23CC(NC(C(CC)N(C)C)=O)(C2)C(C)O3)cc(N)cc(C)c1F C(=O)(CCCCCCN=[N+]=[N-])NC1C(OC)CN(C(c2cc(C)[nH]n2)=O)C1 Cc1cc(C(N2CC(NC(=O)CC34CCCC3C4)CC2CO)=O)cc(C)c1F C1(CC(=O)OC2(CO)CCC(C)C2)CN(C(=O)OC(C)(C)C)CC1(C)C c1(OCCOC)ccc(C(N2CCC(CNC(=O)Cc3nncs3)CC2)=O)cn1 CN1CCN(C(=O)C(CCF)NC(=O)C=C2CCCCC2)CC1=O C(=O)(CCCC(F)(F)F)N(C(C)CCNC(=O)Cc1ccccn1)C C(=O)(CC1=CCCC1)N(CCC(=O)N1CC(C(O)C=O)C1)C.C(CC(C)(C)C)N CC(CNC(c1c(F)cc(F)c(F)c1F)=O)N=c1[nH]c2ccc(O)cc2s1 CN1CCOC(C(N2CCCC2CN(C(=O)C=CCN2CCCC2)C2CC2)=O)C1 c1(CC)ccc(F)c(C(=O)NCC(CC(C)C)NC(C2(Cl)CC2(C)C)=O)c1F Cc1ccnc(C(=O)NC23CCC(NC(=O)Cn4ccnc4C)(CC2)C3)c1F N1(C(c2ccc(Cl)cc2)=O)CCCC2(C1)CN(C(=O)C(F)(F)C1CCOCC1)C2 C1(C(N2C(CNC(C3C(c4onc(COC)n4)C3)=O)C=CC2)=O)CC2CCC(C1)O2 c1(C(N2C3(CNC(C(CC)CO)=O)CC(C2)C3)=O)ccc(O)cc1C(F)F c1(C(N2CC(O)(CNC(C(C)Cn3cccn3)=O)C2)=O)cnccc1Br C#Cc1ccc(C2(C(=O)NCC3(O)CC(CNC(C4CC5CC5C4)=O)C3)CC2)cc1 N1(C(c2n(C)cc(Br)c2)=O)CCC(NC(c2ccnn2C(F)F)=O)C(O)C1 C#CCC(CC(F)F)C(=O)N1CCCC(C(=O)N(CC2=CCSC2)C)CC1 C1(CCCNC(=O)C=CC2CCOC2)CCCN1C(=O)CCc1cncnc1 c1(SC)cnccc1CCNC(=O)NC(c1nccn1C(F)F)C C1(NC(C(C2CN(C(CCOCCC)=O)C2)O)=O)COCC1C1CC1 C1(NCCC2CCCC(C)C2)CCC(O)CNC1 c1(CCC)onc(C)c1C(N1CCN(C2CCCN(C(=O)CC3CC3)C2)CC1)=O c1(CCC(N2CC(N(C(=O)CCCF)C)C(C)(C)C2)=O)nc2cccnc2[nH]1 CC1CN(C(c2ccc(Oc3cccc(Cl)c3)cc2)=O)CC1NC(=O)CCF c1(Cn2cc(C3(NC(Cn4ncc(CC)c4)=O)CCC3)nn2)cc(F)ccc1F c1(CC(=O)NC(CCCC)CNC(=O)CCCCOCC)ccc(OC)c(F)c1 C1(CCCNC(C=CC)=O)CCN(C(C2(CF)CC2(F)F)=O)CC1 c1(NC)ccc(C(=O)NCCCC(C)NC(=O)C(O)CF)cc1F C(=O)(C(C)CN(C)C)NCCCN(C(=O)C(C)(C)c1cscc1Cl)C(C)C N1(C(c2oc(CC)c(C)c2)=O)CC2(CCN2C(C2CC=CCC2C)=O)C1 N1(C(CC2OCCN(C(c3ccn(C)c3)=O)C2)=O)CCN2CCCC2C1 c1(C(=O)NC(C(C)(C)NC(CCCCOCCC=C)=O)C)cc2c(s1)CCC2 c1(CC)cc(C(=O)N(CC(C)NC(C2CCC(N(C)CC)CC2)=O)C)ccc1C C#Cc1cccc(C(=O)N(C(C)CNC(=O)Cn2cc(Cl)cn2)CC)c1F [N-]=[N+]=Nc1ccccc1NC(C1COC2(C1)CN(C(=O)Cc1ccsn1)C2)=O C1(COC)CNC(CNCCCC2CCCC2)C1 Cc1scc(C(=O)NCc2cnn(C)c2C(=O)NCC2(CO)CCC2)c1C Cc1c(NCC(=O)NCc2ccsc2Cl)ncnc1NC1(CO)CCC(C)C1 CCC(C)CN=c1cccc(S(=O)(=O)NC2(C(c3ccccc3)=O)CC2)[nH]1 c1(C(=O)NC2CN(C(=O)CCn3cnnn3)C3CC23)cccc(Cl)c1Cl c1(C2(OC)CCC2)c(F)cccc1F.C12(OC)CN(C1)C(=O)C2 Cn1cnn(CCC(=O)NC2COCC2n2cc(CC(O)C3CC3)nn2)c1=O c1(C(=O)OCC)sc(C)cc1NC1(c2nnnn2C)CCCC1C N1(C(CN(CCOC)C)=O)CCC1(C)CCC(=O)NCCCCSC N1(C(CC=CC)=O)CCC2(CCCC2NC(=O)C(C)CCOC)CC1 N1(C(c2c(C(C)C)c[nH]c2)=O)CCCC(CN(C(=O)C(C)OCCN(C)C)C)C1 N1(C(CN(C)CC)=O)CCCC(COC)(NC(c2ccc(-c3cc[nH]n3)s2)=O)C1 C1(COC)(NC(C2CC23CCOC3)=O)CCN(C(=O)Cc2cnc(C)s2)C1 c1(C(=O)NC(CN(C(CN(C(C)C)C)=O)C)C)cc(Br)c2[nH]cnc2c1 C12CC3CN(CC3C1)OC2=O.CCC(O)(Cn1nnnc1-c1ccccc1)CC c1(-c2nc(NC3CCC(NC(CCCC#C)=O)C3)sc2)cc(C)cc(C)c1 N1(C(CC2CCC(=O)CC2)=O)CCC(C(N2CCCCC2CF)=O)C12CC2 C(c1ccc(Cl)cc1Cl)=CC(N1CC(OC)CC(NC(C=CSC)=O)C1)=O CC(C)CC(C(=O)C(=O)C=Cc1ccsc1)ONC(=O)C1CC(C(C)(C)O)C1.N N1(C(C(CC)OC)=O)CC(NC(c2cc(OC)nn2C)=O)CC12CCC2 S(=O)(=O)(c1c[nH]ccc1=NCc1cc(Cl)on1)NCC(C)n1cncn1 C1(NC(c2ccc(CO)s2)=O)CC(CNC(C2(O)CCCC2)=O)C(O)C1 c1(CCC(=O)NC(CNC(C(C)SCCCC)=O)(C)CO)csc2ccccc12 CC1CN(C(=O)CCC2(C)CC2)CCCN1C(=O)CCC1CCC(=O)C1 CC1CCC(NC(=O)CCc2cccc(O)n2)CN1C(=O)C1=CCCOC1 Cc1cc(CNC(C2CN(Cc3ccc(Cl)cc3F)CCO2)=O)cc(C)c1F c1(N2CCC(NC(=O)NC3C(C(C)(F)F)C3)C(F)C2)ncnc(Cl)c1[N+](=O)[O-] c1(-c2ccc(C)o2)nc(C)c(C(=O)N(CCNC(C2CCCSC2)=O)C2CC2)s1 c1(C(=O)NCCN(C(CN(S(CC)(=O)=O)C)=O)C(C)C)csc(S)n1 C12(C(=O)NCCOC3CN(C(CC(C)F)=O)C3)CCOC1CCOC2 c1(NC2CC3CN(C(=O)OC(C)(C)C)CC3C2)nccc2c1NCCC2 N(C1c2ccccc2CC1NC(=O)CC(C)(C)N(C)C)C(CSCC=C)=O c1(NC(c2nc(O)n[nH]2)C)nc2cc[nH]c2c(=NCC2CC(=O)NC(C)C2)[nH]1 CCC(C)CCC(=O)NC1(CCNC(C2COCCOC2)=O)CC1 C(CCCC(=O)N1CC2CC2(CNC(c2coc(C(F)(F)F)n2)=O)C1)OCC C1CCCC(N=c2[nH]ccn3nnnc23)C1.Cc1cc(Cl)cc(C)c1C=O N1(C(CCC=CC)=O)CCN(C(=O)C(C)C2CCCO2)CC1CCO c1(C(=O)NC2C=CCN(C(C(CC)(F)F)=O)C2)ccnc2c1CCC2 c1(NC(=O)N(c2ccccc2Cl)CCN(CC(F)(F)F)C)ccc(=O)n(C2CC2)c1 CC1=C(C(=O)NCC2CCCCC2NC(c2cc(F)n[nH]2)=O)CCC1 N1(C(C2=CC(C)C2)=O)CCC2(C1)CN(C(=O)Cc1nc[nH]n1)CCO2 Cc1conc1C(=O)NC1(CCNC(c2snnc2C(C)C)=O)CC1 c1(NCCN(CCOCCC)C)cc(=NC2CCCN(C(C)C)C2)[nH]c(COC)n1 CC1CN(C(c2snc(O)c2Cl)=O)CCC1NC(=O)CN1CC(=O)N(C)C1=O C#CC1(CNC(=O)Nc2ccc(CNCCCC)cc2)CCCC1 N1(C(C(C)(C)N=[N+]=[N-])=O)CCCCCCC1C(=O)NCC1CCCCC1O C1(C(=O)NC(CCCCNC(CCC#CC)=O)CO)Cc2ccccc2C1(C)C C1(C(=O)NCC2N(CC)CCC2)CC2C=CC1N(C(=O)CC1CC(C)(C)CO1)C2 c1(C(N(CCCNC(C2OCC(C)C2)=O)C2CC2)=O)ccnc(S)c1 c1(C(N2CC(SCC(N3CC(C)NCC3)=O)OCC2)=O)nccc2c1NCCC2 C1(CC(=O)OCC)CC2CCC(C1)N2Cc1cc(-c2ccccc2)cn1C N1(C(C(Cn2cccn2)NC(C=Cc2cc(C)no2)=O)=O)CCC(F)C(F)C1 N1(C(CC2N(C(COC(CC)(C)C)=O)CC(C)(C)C2)=O)Cc2ccnn2CC1C C1(C(N2CC(NC(C(C(=O)OC)C)=O)(CO)C2)=O)CCCN1S(=N)(=O)N(C)C C1(COC)CN(C(=O)CC2CC=CCC2)CCN1C(=O)C(C)=CC1CC1 CC(=O)CCCC(C)C(=O)N(C)CC1CCCCN1C(=O)CC1CCC(=O)N1 C=CCCCC(=O)N(C)CCOCCN(C(=O)C(F)(F)CN(C)C)C N1(C(C2(COC)CCCC2)=O)CCC(C)C(CNC(c2c[nH]nc2[N+](=O)[O-])=O)C1 N1(C(C(CCN(C)C)NC(C2CN(C)C2)=O)=O)CCC(N=[N+]=[N-])C1 C1(OCC(=O)OCc2cocn2)CC(=O)C1 N1(C(C)C2CC2)CCC(CNc2cncc(-n3cccn3)n2)CC1 C1(NC(C23CC(C)(C2)C3)=O)CCN(C(C2(c3ccc(Cl)cc3)CCCC2)=O)CC1O C1(CCNC(C=CCN(C)C(C2(C)CCCS2)=O)=O)CCCC2CC12 C(N=c1[nH]c(=NC2CCCC2N2CCCCC2)c2[nH]ccc2[nH]1)c1ccc(Cl)o1 C(=O)(C(N=[N+]=[N-])C(C)C)N1C(CC(=O)NC(CC=C)CC(F)F)C2CCCC21 Cc1cocc1C(=O)NC1CCC(N(C)C(C23CC(CO2)C3)=O)C1 CC(c1ccccc1)=CC(N1CC(CNC(=O)C(C)OCOC)C(O)C1)=O C(=O)(C1=CCC(C)CC1)N1CCC(=C)CC1C(N1CC(c2cc(O)n[nH]2)C1)=O c1(C(=O)NCCN(C(C(c2c(C)cccc2)C)=O)C)noc2c1CC(C)CC2 C(=O)(C1=CS(=O)CCC1)N1CCCCC(NC(c2cc(CC)[nH]n2)=O)C1 Cc1cc(CNC(N2CCOCC3(COC3)C2)=O)c2c(c1)CCC2 N1(C(C2(CSC)CC2)=O)CCCC2(CCC(NC(c3cc(SC)c(C)o3)=O)C2)C1 N1(C(C2C(C)(C)CCN2C(=O)CC2=CCCC2)=O)CC2(CCOCC2)C1 CC=C=CCCN=c1[nH]c(=NCCCCN(C)C2CC2)[nH]c2c1CCC2 N1(C(C2(OC)CCN(C(C(CC#C)O)=O)C2)=O)CCOC2(CC2)C1 N1(C(=O)OC(C)(C)C)CCC2CCC12C(=O)NCCCCOc1ccc(F)cn1 c1(CC(C)NC(=O)N(c2ccc(Cl)nc2)CCO)ccccc1C(F)(F)F n1(Cc2cccc(CNC(c3c(Cl)cnc(C)n3)=O)c2)c(=O)n(C)c2ccccc12 S(=O)(=O)(c1cccnc1N(C)C(c1ccc(Cl)cc1)C)NC(c1c(C)ncs1)C Cc1cc(F)c(F)cc1NC(c1cscc1-c1nccs1)=O CCCC(C)C(=O)N(C(C)(C)CC(=O)N(C1(C)CC1)C)C N1(C(CCC=CC)=O)CCN(C(=O)Cc2occc2C)C(CCOC)C1 N1(C(CC(C)OC)=O)CCc2ccccc2C1CNC(c1cncc(Cl)c1Cl)=O C1(NC(C=C(C)C(F)F)=O)COCC1OC(C)C=CC(=O)N(C)C C1(C(=O)OC)CN(C(=O)NCc2c(Cl)cnc(F)c2Cl)CC(F)(F)C1 C1(N(C(=O)CCOCCCNC(c2cncc(O)c2)=O)C)CCC(CO)CC1 Cc1cccc(CNC(c2ccc(-c3c(O)cccc3F)nc2)=O)c1Br C(=O)(CCCC(=O)N1CCC(CNC(=O)Cc2ccnc(Cl)c2F)C1)OC C(=O)(CCCCC(N)=O)N1CC(N2CCN(C(C=NOC)=O)CC2)C1.C(=O)OC CN1CCCN(C(=O)C2=CCC(NC(=O)CCN(C)C)C2)CC1=O CN1CC(C)(C)CC1C(=O)NC1CCC(C(=O)NOCCN2CCCC2=O)C1 C(CNC(C1CCOC1)=O)(CC(=O)NCCSC(F)F)OC N1(c2n(CC=C)c(CC=C)nn2)CCC(C(=O)OC)C1C C1(CNC(c2c(OC)nsc2)=O)(NC(C2CC=CCC2)=O)CCC(C)(C)CC1 C(=O)(CC(C)(C)C(C)(F)F)N1CCN(C(C=C(COC)C)=O)C(C2CCCC2)C1 CC(C(C)(O)C(=O)N1CCC(C)(NC(c2cc[nH]n2)=O)C1)c1ccccc1 c1(C(=O)NC2(CNC(c3cc(CCOC)on3)=O)CC2)n[nH]c2ccc(O)cc12 c1(C(=O)NC2C(NC(CCNC(C)=O)=O)CCCC2)cccc2ncnc(O)c12 C=CC(C)(C)CC(=O)NC1(CN(C)C(C2CCN(CC)CC2)=O)CC1 C1(NC(CCOC)=O)(CO)CCN(C(C2(c3cccc(C(F)F)c3)CC2)=O)C1 C1(NC(c2c(C)coc2)=O)CC(C)CN(C(=O)CCc2cccc(Cl)c2)C1 C1(c2n(C)ccn2)CN(C(=O)C=CC2CC2)CCN1C(C1CC2COCC2C1)=O c1(C(=O)NCC2C3CN(C(=O)CC(F)F)CC23)ccc2c(c1)CCCS2 c1(C(=O)NC2C(NC(CC3C(CC)C3)=O)CCC2)cccc(N2CCOCC2)c1 c1(CCC(N2C(C3CCN(C(CCC=C)=O)C3)CCC2)=O)ccc(OCC)cc1 C1(NC(C(C(C)C)c2ccccc2)=O)CCCCN(C(=O)C=Cc2ncco2)C1 CC(C(=O)NC1C2CCC1N(C(c1ccc(OC3CC3)cc1)=O)C2)S(N)(=O)=O C1(CNC(c2c(Br)cn(C)c2)=O)CCC2(CCN(C(=O)CC=CCF)CC2)O1 N1(C(c2c(C(N)=O)cccn2)=O)CC2CCC(C1)N2C(=O)Cn1ncccc1=O C1(NC(C(C(C)(F)F)F)=O)CCCC12CCN(C(C1(CO)CCCCO1)=O)CC2 CC(C)(C)C(=O)CCC(=O)N1CC=CC(C(=O)NCC2(C)CC2)C1 N1(C(c2c(OC)cc(C)s2)=O)CCC2CCN(C(=O)CCCC(C)C)C2C1 C1(NC(C2(COC)CCOC2)=O)C=CCN(C(c2ccc(C3CC3)s2)=O)C1 c1(C(=O)NCC2C(NC(c3cc(C4CCCCC4)[nH]n3)=O)CC2)c[nH]c(Br)c1 C12(NC(=O)Cc3c(F)cncc3Cl)CCCC1CN(C(c1cc[nH]n1)=O)C2 c1(C(=O)NC(CN(C(CN(CCC)C)=O)CC)C)cc(C)n(C(CC)CC)n1 C1(NC(N(C2CCCC2)CC(=O)NCC2=NOCC2)=O)C2CCC3C(C2)CC13 N1(C(c2c(C(C)C)con2)=O)CCC2(CC2NC(c2cn3ccsc3n2)=O)C1 C(=O)(C(CC)C(C)O)N(CCN(C(=O)C=Cc1cncc(O)c1)CC)CC c1(C(=O)NCCCNC(=O)CCC2CCCCO2)ccc(F)c2ncccc12 N1(c2c(C(=O)OC)nccn2)CCCC2(NC(=O)Cc3sccc3C)CC2C1 c1(OCC)cc(C(N2CC3C(C(=O)N(C)C(c4nocc4C)C)C3C2)=O)ccn1 CCCC(C(=O)N1CCC(C(=O)N(CC(O)COCC)C)(COC)C1)OC CC(C(C)C(=O)NCCc1ccccc1F)NC(=O)CCn1ccnn1 N1(C(COC2CC(NC(C(C)C#N)=O)C2)=O)CC(O)CC1(C)C1CC1 c1(OC)nc(Cl)ccc1C(N1CCC(NC(C2(C3CC3)CCCO2)=O)C(F)C1)=O N1(C(CSCCOC)=O)CCCC12CCN(C(=O)CCc1cn(C)nn1)C2 N1(C(c2cc(CC)ncn2)=O)CC(C(=O)NCCN2CCC(CO)C2)C2(CC2)C1 C1(NCC2CC(C)OCC2)CCN(C(=O)C(C)S(N)(=O)=O)CC1C C1(C(N(CC(C)NC(C23CC2CNC3=O)=O)CC)=O)CCC2(CCC2)C1 N1(C(c2ccn(C)c2)=O)CC2(CCN(C(C3CCCN(CC(F)F)C3)=O)C2)C1 Cc1ccc(N(S(=O)(=O)c2cnsc2)C2CCCC2)c([N+](=O)[O-])c1 C1(CNC(c2ncn(C)n2)=O)CC2CC1CN2C(=O)C(F)(F)c1nccs1 C(=O)(C1=CS(=O)CCC1)NC12C(NC(c3cc(OC)n[nH]3)=O)CC(CC1)C2 C1(CC(=O)NCC(c2ccc(F)cc2)NC(c2c(C)ncs2)=O)CC2(CC2)CO1 O=C(C1=Cc2ccccc2C1O)NCCCNC(c1ccoc1C1CC1)=O c1(C(=O)NC(C(=O)NCCC(C)(C)O)Cc2cn[nH]c2)c(F)cccc1F C(=O)(C1=CCCCC1C)N1C(C(=O)NCCC(=O)OC)CCC1C(C)C c1(CCC(=O)NCCCCNC(C2C(CC)OCC2)=O)cccc(C#N)c1 c1(C(=O)NCC2CC2C(=O)NCCC2(O)CCC2)cccc(Cl)c1Br.CO.N C(CCCCC(=O)NC12COC(CNC(C3CC3OC(C)(C)C)=O)(C1)C2)OC C1(NC(c2cc(C(C)C)nn2C)=O)CC2CC1N(C(c1cc(=N)[nH]n1C)=O)C2 C1(CCNC(CN(C(=O)C(O)CN(C)C)C(C)C)=O)CCC(C)(C)C1 Cc1c(C(=O)NC2C3CC2N(C(=O)CN2CCCCC2C)C3)nn(C)c1Br O=C(CC(F)(F)Cc1ccccc1)NCC1CCCN1Cc1ccc(F)cc1Cl C1(C(N2CCN(C(CS(N)(=O)=O)=O)C(CCO)C2)=O)CCOC2(CCCC2)C1 N#Cc1cn[nH]c1C(=O)NC1CC(CNC(=O)CCCc2ccccc2)C1 C(=O)(CCC(C)(F)F)N1CCC(C(NOCCC#C)=O)C1C(C)C c1(C(N(C2CCN(C(C34CCN(CC3)C4)=O)C2)CC)=O)[nH]cc(CC)c1C N1(C(C2N(C)SCC2)=O)CCC(Cn2cc(-c3cnc(C)o3)nn2)C1(C)C Cn1ncc(Cl)c1CC(=O)NC1CCCC(NC(=O)CC(=O)OC(C)(C)C)C1 c1(C(N(C)CC2CCN(C(c3cnc(O)c(F)c3)=O)C2)=O)cc2scc(Cl)c2[nH]1 C1(NC(c2nc(C(C)(C)C)oc2)=O)CCC2CN(C(=O)C=Cc3cnc[nH]3)CC2C1 c1(C(=O)NCCCN(C(c2n(C=C)nnc2)=O)C)cc(OC)cc(OC(F)F)c1 c1(C(N2CC(C(=O)NCC(=C)C)(CC)C2)=O)ccc(OCCC(C)C)cc1 Cc1nc2c([nH]1)CN(C(=O)C(C)(C)CCNC(=O)CCCn1ccnc1)CC2 CC12CN(C(C34CCC(C3)OC4C)=O)C(C(N3CCOC(C4(C)CC4)C3)=O)(C1)C2 C1(C(=O)NCC2C(CC(=O)NCCC(C)F)C2)CCOC1C Cc1ccc(C(F)F)cc1C(=O)NC1CCC1NC(c1cnc(C(C)C)s1)=O c1(OCC(=O)NC(CC(C)C)CNC(=O)C=C2CC2)ccc(F)cc1O c1(C2(C(=O)NC3C(CNC(c4cccc[n+]4[O-])=O)COC3)CC2)ccc(F)cc1 N1(C(c2c(CC)c[nH]c2)=O)CC2CC(NC(c3ccc(S(N)(=O)=O)s3)=O)C(C2)C1 CC(C)C(C(=O)NCC1CCN1C(c1cncn1C)=O)n1ncc(N)n1 C1(C(=O)NCC(CN(C(c2ccc(C)o2)=O)C)O)CC12CCC(=O)CC2 C1(NC(c2ccc(CC)[nH]2)=O)CCCCCC1C(=O)N(C1CCOC1)C c12cc(nn1C)CNC2=O.C1(c2ccccc2)(CC(=O)N(C)C)CCCC1 N1(C(C=Cc2n(C)ccc2)=O)CCC(NC(c2ccc(O)cc2Cl)=O)C(O)C1 N1(C(CC#N)=O)CCC2(CCC2)C(CNC(=O)CSc2ccc3c(c2)CCC3)C1 C1(CC)CN(C(=O)C=Cc2ncc[nH]2)CCN1C(=O)CN(C)CCOC(C)(C)C C1(NC(c2cc(CCC)[nH]n2)=O)C2CC3C1C3C2C(=O)NC(C)CO c1(C(=O)NCC=CCNC(C2C(CCC)(CO)C2)=O)occc1C(C)C CCCCCCC(C)CC(=O)N1CCC(C2CC2)(CNC(=O)CCC(C)(C)O)C1 C1(OC)CCCC(C(=O)N(CCCCCNC(=O)CSc2n[nH]c(C)n2)C)C1 c1(C(C(=O)NC2(C)CN(C(=O)COCC3CCOC3)C2)OC)ccc(Cl)cc1 c1(C(=O)NC2CN(C(c3ccc(CC)s3)=O)CC2C)cccc(S(N)(=O)=O)c1 c1(C(C(=O)NCCC2(C)CC2)N(C2COC(=O)O2)CCOC)c(SC)cccc1F c1(C(C(=O)NC(CC)C)N(C)CCc2cnn(C)c2)ccc(C(C)(F)F)cc1 C12CN(C(C)(C)C1)CC(=O)NS(=O)(=O)C2.Cc1nc(O)c(C(=O)O)s1 c1(C(=O)NCCC(=O)OCC(c2ccc(Cl)cc2)=O)c(O)cc(O)cc1O C(CN=c1nc(N2CCOC(c3cn[nH]c3)C2)c2c([nH]1)CCOC2)N(CCC)C c1(C(C)N(C)CCOCCNC(C2CC3CC3C2)=O)cc2ccccc2o1 N1(C(C2CC(C)(F)C2)=O)CCC(C(F)(F)F)C(NC(C2CCOCC2)=O)C1 C(N=c1nc2sccc2c(N2CCC3(CCCC3)C2)[nH]1)C1C(C)CCCC1 C(=O)(C(F)C=O)OCCl.N1(C(C)(C)C)CC2C(C1)N2C(=O)CC1C2COCC12 CCC(C)(C(=O)NCC1(F)CCC(NC(c2nccc3n[nH]cc23)=O)C1)C(F)F N1(C(C(c2ccccc2)SC)=O)CCN(C(=O)CC(F)F)CC1C C1(CCC)(NC(=O)CN2C(=O)CNC2=O)CCCN(C(=O)CS(N)(=O)=O)C1 C1(CNC(CSC)=O)CN(C(=O)Cn2cccn2)CC(C)(C)O1 N1(C(C2C(OCC)C2)=O)CCCC12CCN(C(c1cn[nH]c1)=O)C2 CCCC(C(O)C(=O)NC1CC2CCC1(CO)C2)NC(=O)CCCC1CCC1 CCCCC(CC)CC(C(=O)NCC(C)C)N(CC)Cc1occc1C O=C(CCCCCCC(=O)NC1CC1)NC1CC1(Cl)Cl C1(CNC(C2CC(=C)C2)=O)CC(C(F)(F)F)CCN1C(=O)C=Cc1cncn1C N1(S(CC)(=O)=O)CCCC(C(=O)N(CC(CC)NC(C2C=C(C)CS2)=O)CC)C1 Cc1cc(=NCC2CCOCC2)[nH]c(NCC2CCCC2C(C)(C)C)n1 C1(CCN(C(c2c(CC)nc[nH]2)=O)C)CCN(C(C2CCN(C(C)=O)C2)=O)CC1 C(CC(O)C(=O)N1CC(CC(F)(F)F)C1)NC(c1n(CCC)ncc1)=O CN1N=C(C(=O)N2CCOC(C(=O)NCCn3cnc(CO)c3)CC2)CCC1=O Cc1ccccc1C(N(C(=O)C=C(Cl)Cl)CC(N1CCCCC1C1CCC1)=O)=O c1(NC(C)=O)ccccc1NC(=O)N(C)CC1CC2CNC1C2 c1(C(N2CCC(NC(CCC#CC)=O)(CO)C2)=O)cc(C)c(C)nc1C N1(C(C2(C)CC2(F)F)=O)CC2CN(C(c3cncs3)=O)CC2C1 C(=O)(C(C)CCCC(C)C)NC1CCN(C(C2CC(CC)OCC2)=O)CC1(C)C N1(C(c2cn(C)nc2)=O)CC(CNC(c2cnn[nH]2)=O)C2(CCOCC2)C1 N1(C(C2(OC)CCSC2)=O)CCC(C2(O)CC(NC(C3CCC(=O)N3)=O)C2)CC1 c1(OC)ncc(C(=O)NC2COCCC2NC(=O)CCNC(c2ccsc2)=O)cn1 CCCC(C(=O)N1CC(O)(C2CCCN2C(=O)C=Cc2ccco2)C1)NC(C)=O C1(CNC(C2CC(NC(C3COCCO3)=O)C(O)C2)=O)CCC2(CC1)CC2 C(=O)(C(F)C(C)C)N(CCOCCNC(C1(CCOC)CCC1)=O)C Cc1cc(C)c(CC(=O)Nc2cccc(NC(C3CC4(CC4)C3)=O)c2)c(C)c1 Cc1cccc(C(=O)NCCC2CC(NC(=O)Cn3cc(CO)nn3)C2)c1F C1(NC(C2CC(CC)C2)=O)CCN(C(=O)C(C)(C)S(C)(=O)=O)CC(C)(C)C1 c1(C(N2C(CC)C(NC(=O)Cc3ccn(C)n3)CCC2)=O)c(C)nc2sccn12 Cc1nc(C(N2CCOC(CCNC(C3CCN(C)C3=O)=O)C2)=O)cc(O)n1 c1(C(N2CCCCC(NC(=O)C=CC=C(Cl)Cl)C2)=O)ccc2scnc2c1 c1(C(=O)NC2C(SC)CN(C(=O)Cc3scnc3C)C2)ccc2[nH]c(=N)[nH]c2c1 C1(NC(=O)CC2CSCCN2C(=O)CC2CSCCO2)CCCC2(C1)N=N2 C1(C(C(=O)N(CC=C)C)(C)C)CCN(C(c2nnsc2C)=O)CC1 C(=O)(CCCCCC(C)O)NC(C1N(C(c2nc(CC)oc2C)=O)CCC1)(C)C c1(C(=O)OCC)cc(C(C(=O)NCCSC)N(C)Cc2ccccc2)on1 c1(C(=O)NC)cccc(NC(C2COCCN2Cc2cc(Br)ccn2)=O)n1 c1(CC)cc(C(=O)NCC2CC3(CC3)CN2C(C2CCCOC2)=O)ccc1Cl N1(C(C(C)N(C)C)=O)CCC2(CC1)CN(C(=O)CCCCCF)CCO2 c1(C(N2CCC(N(C)C(c3cc(Br)cnc3Br)=O)C2)=O)c[nH]c2ccc(F)cc12 S(=O)(=O)(c1cccnc1NC(c1cn(C)nn1)C)N1CCCC(C(=O)NCC)C1 n1(C(CC)(C)C)nnnc1C(c1cnc(C)s1)NCc1nc(Cl)cs1 c1(C(=O)NC(C2(O)CN(C(Cc3c(C)nsc3)=O)C2)C)ccc2sccc2c1 CC1CCc2sc(C(=O)N(CCCOCCNC(C3(C)CC(F)C3)=O)C)cc2C1 C1(CC(=O)N(CC(C)NC(=O)CCc2nncs2)CC)COCCN1CC(F)F C1(C(=O)NC2C(CNC(c3cn(CCCC)nn3)=O)CCC2)CCC(=O)N(C)C1 N1(C(CC2C(C)(C)C2)=O)CCC(CCCCNC(=O)C=CC=C(Cl)Cl)CC1 CCCCC(C(=O)N1CCCC(F)(C(=O)NC2CC(=O)N(C(C)C)C2)C1)N(C)C N1(C(c2cc(CC)nnc2C)=O)CCCN(C(C2CCC2C(C)(C)C)=O)C(C)C1 S(=O)(=O)(c1ccccc1F)NC1CCCN(C(c2ncn(C(C)C)n2)=O)CC1 C(=O)(C(CC(C)C)N1CCCCC1=O)NC1CN(C(CN(C)CC)=O)C1 CC(CCC(=O)NOCC(N)=O)NC(=O)Cn1cncc1C(C)O N1(C(c2c(CCC)nns2)=O)CC(NC(=O)C(C)CO)CC2(CCOCC2)C1 C(=O)(C(CO)C(F)(F)F)N1CCN(CCCNC(C2(C)CCC(C)C2)=O)CC1 c1(C(=O)NC(CC)CNC(C2(C)CCCS2(=O)=O)=O)cc(N)c(F)cc1C C1(C)(NC(C2(CC)CCNC2=O)=O)CCCN(C(c2ccc(C3CC3)cn2)=O)C1 c1(C(=O)NCCN(c2ncnc(N(C)C)n2)CCC)ccc(F)c(Cl)c1 c1(NC(C)=O)ccc(C(=O)NC2CC2C(N2CCN(C)CC2)=O)c(C(F)(F)F)c1 C=CCC(C)(C)CNC(c1nnnn1C(C)C)CCOC c1(C(=O)NC2C(NC(c3cc(OC)oc3C)=O)CCOC2)cnn2ccccc12 C1(CNC(=O)Cc2ccc(Cl)cn2)CC2CCC(C1)N2C(=O)C(O)c1ccsc1 c1(C(=O)NC2CC(C)CN(C(=O)C(O)C(F)(F)F)C2)c[nH]c2ccc(F)cc12 c1(C(=O)NC2CC3(C2)CN(C(c2cc(Br)c[nH]2)=O)C3)cccc2c(Br)cccc12 N1(C(C23CC(C)(C2)C3)=O)CC2CC(NC(c3cscc3C(N)=O)=O)CC2C1 C1(CNC(c2n(C)c(S)nc2)=O)CC12CCN(C(=O)C(O)C(F)F)CC2 c1(C(=O)NCC(CNC(C2CCC(F)(F)CO2)=O)OC)c(F)cc(F)cc1F n1(CC(=O)NC2CN(C(c3nc(C)oc3)=O)C3C2C3)cc(Cl)c(O)nc1=O c1(C(=O)NCC2N(C(c3ccc(C#C)o3)=O)CCC2)cnn2c1N(C)CC2 S(=O)(=O)(c1cc(Cl)ccc1Cl)NCCC(=O)NC(C(=O)OC)CSC c1(OC)cc(Br)ccc1CN1CCOC(CNC(c2cc(F)ccc2O)=O)C1 O=C(C(CO)C(F)(F)F)N1CC2CC2C1C(=O)NOCC=CCl C#Cc1cc(C(N2CCCC2CN(C(=O)C(CC)NC(N)=O)C)=O)cc(Br)c1 CCCCS(=O)(=O)CC(=O)NC1(CN(C)C(C2CC2CN(C)C)=O)CC1 n1(C(c2c(OC)ccc(Br)c2)=O)ccc(=O)n(C)c1=O C1(C)(NC(c2c(C)cc(C)[nH]2)=O)CCN(C(c2cc(Br)cn2C)=O)CC1 Cc1c(C(N2CC(NC(=O)COCc3nccn3C)CC(O)C2)=O)cccc1F C1(OC)CS(=O)(=O)CC1NCCN(C)CCSC CC1COCCC1N(C)C(c1cccc(CO)n1)=O.c12nnn(C)c1CNC2=O c1(C(=O)NC(CCNc2cn(COC)nc2)C)ccc(F)cc1O N1(C(c2ccc(S(N)(=O)=O)cc2)=O)CC2CC(N=c3ccnc(CO)[nH]3)C2C1 NS(=O)(=O)c1ccc(NC(c2nnnn2C2CCC2)C2CC3CC3C2)cc1 c1(C(=O)NC2C(CNC(c3cn(C)c(=O)nc3O)=O)C2)ccc2c(c1)C(=O)NC2 C1(NC(Cc2nc(C)[nH]n2)=O)CCCCN(C(=O)C(N2CCC(C)C2)=O)C1 C1(NC(=O)Cc2cnsc2)CC2CN(C(c3ncc(F)cc3F)=O)CCN2C1=O C1(C(C)C)CCC(NC(=O)C(C2CCCO2)C2CC2)CC1 c1(CNC(=O)OCCOC(c2c(N(C)C)nn(C)c2)=O)cnc(O)c2ccsc12 c1(N(C(C(=O)NC)C2CC2OC)CC)nc(Oc2ccc(OC)cc2)cc(C)n1.CC c1(OC)ccc(CC(=O)NCCN(C(=O)CCS(=O)(=O)N(C)C)C)c(C)c1 Cc1ncccc1C=CC(=O)NC(C)(CNC(C1CCOC1)=O)CO C(=O)(C(O)C(F)(F)F)N1CCC(NC(C2CC(F)(F)C2(F)F)=O)CC1 C12(CNC(c3n(C)ncc3Cl)=O)CCC1CN(C(=O)CC1(n3ccnc3)CC1)C2 C12(CN(C)C(=O)NCc3cscc3Br)CC(F)C1C2 C(CC(F)F)(C(=O)N1CCOC(C(=O)N(C)C)C1)NC(CC(C)F)=O c1(C(=O)NC2(C)CCN(C(c3c(CC)nn[nH]3)=O)C2)cnc2c(F)cccc2c1 C1(SC)CN(C(=O)C(C)O)CC1CNC(=O)C(C)(C)C C1(C2CC2)(CNC(=O)C=C(Cl)Cl)CCN(C(=O)CCN2CCCS2(=O)=O)C1 c1(C(=O)OC)cc(Br)c(F)cc1N(C1CCNCC12CC2)C(=O)COC(C)(C)C C1(C(=O)NCC2(CO)C(C=C)C2)CC2CCC(C1)N2C(c1c[nH]nc1CC)=O c1(C(c2ccsn2)NCC(COCC)OC(C)=O)nnnn1CCC.C(C)(C)(C)O C1(C(=O)NCCCN(C(=O)CC2CCC(=O)N2)C)CCc2nccn2C1 c1(C(=O)NC(CC)(C)CNC(C2CCCCC(=O)N2)=O)cc(F)c(C)cc1Cl CON(Cc1ccc(C)o1)C(=O)C(CCOC)NC(=O)CC1CCCC2CC12 C=CCCC(C)(C)C(=O)NCC(CC(=O)N1CC(CO)(CF)C1)OC c1(OC)cc(C)ccc1C(N1CC(NC(c2cnn(CCF)c2)=O)CC1C)=O S(=O)(=O)(c1ccc2c(c1)OCCO2)N1Cc2c(-c3c(C)csc3)n[nH]c2CC1.C C(=O)(C1Cc2ccccc21)NCc1nccc(-n2cc(C)c(=N)[nH]2)c1 N1(C(C(C(CC)C)OC)=O)CC2(NC(c3scc(C)c3C)=O)CCCC2(F)C1 N1(C(CCCSCC)=O)CC(CC(C)NC(C2CC2(C)C)=O)C1 C#CCC(C)(C)C(=O)N1CCC(NC(=O)NCC23CCCC2C3(F)F)C(F)C1 CC1C(NC(=O)C2=C(Cl)CCOC2)CC2CCC1N2C(C1CCS(=O)(=O)C1)=O Cc1ccc(C(=O)NC2CCC(NC(=O)CCCC(=O)NC(C)C)CC2)c(O)n1 CC1(C)OCCC1(O)C(=O)NCC1CCC1NC(C1(O)CCCCCC1)=O C1(C(N2CC(C(C(=O)NCC3(CCC=C)CC3)O)C2)=O)CC(=O)C1(C)C C1(CNC(CCC2(C)CN(C(=O)CCC(=O)C3CC3)C2)=O)CCC2(CCC2)C1 CCCC(C)CC(=O)NCCCN(C(=O)CN1CCCCCC1)CC C(N=c1ccnc(C)[nH]1)C1CCCC(NC(C(C)OC)=O)C1 CCCC(C)(CC)C(=O)N1CC2CCCC2(C(=O)NOCCC(C)O)C1 c1(NC(C2CCCN(C(=O)CCn3ccnc3)C2)C)ncnc2c1cnn2C C1(C)(C(=O)NC(C2CCCC2)CNC(c2c(CC)ncs2)=O)CC=CCO1 C12CC3CCC(C1)N3C2=O.c1(OC)cc(CN2CCOCC2)ccc1OC(C)=O C1(CNC(c2cnc(C)[nH]2)=O)CN(C(=O)Cn2cc(C(=O)C3CC3)nn2)CCCO1 C1(CNC(=O)CCOC2COC2)CCCC2CN(C(C3OCCO3)=O)CC12 C1(NC(CC2C(C)CCC2)=O)CCOC(C(=O)NCCC2(C)CCCCC2)C1 C12(C(N3CCN(C(CNC(CCC)=O)=O)CC3C(C)C)=O)CC1COC21CCC1 O=C(C1COc2ccc(F)cc21)NCC1(NC(c2ccco2)=O)CCOC1 S(=O)(=O)(c1cccnc1N1CC2CCC(C1)C2CN)SC C1(CC)CN(C(c2cn(C)cn2)=O)CCC1NC(c1sccc1COC)=O C1(C(C(=O)NCCOC)O)CCCC1(C)C.C(C)(C)(C)N(CCOCO)C(C)C1CC1 C(C)(CCC#N)(c1nnnn1C1CCOC1)NCc1ncc(C(C)(C)C)o1 N1(C(CS(N)(=O)=O)=O)CCC2(CCCC2NC(=O)CN2Cc3ccccc3C2)C1 n1(COC)c(CNC(=O)C(C(C)C)NC(=O)COCCCN=[N+]=[N-])cnc1C C1(c2nnnn2C(C)C)(NCc2ccc(OC)c(F)c2)CCCC(C#N)C1 c1(C(=O)NC2CC(C)N(C(c3cc4ccccn4c3)=O)C2)nc2c(s1)CCCC2 c1(CC)cc(C(=O)NCC(CNC(c2ccsc2OC)=O)C(F)(F)F)ccc1C N1(CC)CCCN(C(C2(NC(=O)CCC3CCCC3)CCCC2)=O)CC1=O c1(C(N2CC3CC(NC(C4(C(N)=O)CC4)=O)CC3C2)=O)cccc2nc(O)[nH]c12 Cc1nc2c(o1)CCN(C(C1CC1NC(c1ccc(I)c(F)c1F)=O)=O)C2 C(CCCCC(=O)NCC(C)(C)NC(c1cccc(N)c1)=O)N(C)C.CCN N1(C(Cc2cc(C)on2)=O)CCC(C2CCCN(C(C3CC=CCC3)=O)C2)C1 C1(CNC(CC)=O)COCC2(CCN(C(=O)Cc3nn(C)cc3Br)C2)O1 c1(-c2cn(CCCC(=O)N3C(CC)CCC3)nn2)cc(OC)c(OC)cc1OC Cc1noc(Cl)c1CCC(=O)NCC1CC1NC(=O)C(C)Cc1ccc(Cl)cc1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)C(C)(F)F)cn(C)c1=O N1(C(c2ccn(CCOC)c2C)=O)CCC(C2CC2)(CNC(c2cncs2)=O)C1 C1(CN(C(=O)C(F)(F)c2cncs2)C)CCN(C(=O)C=CC2CCCC2)C1 c1(CNC(C)=O)cccc(C(N2CC(NC(=O)C(C)NC=O)C2)=O)c1 C1(NC(CCC(C)O)=O)Cc2ccccc2N(C(=O)CC2(C)CCCCCC2)C1 C1(N(C(c2ncoc2Br)=O)CC)CCN(C(c2cc(Cl)cnn2)=O)CC1 CCCS(=O)(=O)CC(=O)N1CCCN(C(=O)CN2CCC(C)(O)C2)CCC1 C1(C(=O)NCC2OCC(C(=O)NC(c3ccccn3)(C)C)C2)CC2(CC2)CO1 CN1C(=O)CCC1CC(=O)NC(c1ccccc1)CNC(=O)CCCN(C)C N1(c2c(OC)cnc(Cl)n2)CC2(CCCC2NC(C2CC23CCC3)=O)C1 C1(NC(C23CC(CCO2)C3)=O)CN(C(C2CCN2C2CCCC2)=O)C2CC12 C(C(=O)NCC(C)(C)CCNC(=O)Cc1cccs1)(C(C)(C)C)N(C)C c1(C(N(CCC)CCNC(C2CCCN2C)=O)=O)cc2ccsc2n1C O=C1CCCCC(C(=O)Cn2cc(C3(NS(=O)(=O)C4CC4)CCCOC3)nn2)N1 C1(C(=O)NCC2CC3CCC2O3)CCN(C(=O)Cc2cc(O)nc(O)n2)C12CC2 c1(N2CCN(C(C3CC(CC)(CC)C3)=O)CC2C)nc(OC)c(F)c(C)n1 C1(NC(c2c(C)nc(C)o2)=O)CCN(C)C12CCCN(C(c1cc(Br)co1)=O)C2 c1(CC)c[nH]c(C(N2CCCC2C(C)NC(=O)Cc2cnoc2)=O)c1 CCS(=O)(=O)CC(=O)N1CCN(C(=O)CCCCN(C)C)C(c2ccncc2)C1 CC1CC(O)CN1C(C1CC1NC(c1cccc(C2CC2)c1)=O)=O C12(CNC(=NCCCOC)NCC(C)COC)COCCN1C(=O)OC2 Cc1cc(C(=O)NCC#CCNC(c2cnn(C)c(=O)c2)=O)c(C)c(C)c1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CN(C(c1onc(CC)c1C)=O)CC2CO C12(CNC(COCCOC)=O)COCCN1C(=O)CN(C(=O)C(C1CC1)SC)C2 N1(C(C(CC)(F)F)=O)CC(C(=O)NCC(c2nccs2)C)CCC1(C)C Cc1cc(OC(C)C(=O)NCC2C=CC(NC(=O)CNC=O)C2)ccc1C(C)C C1(C(C)NC(c2coc(C(C)(C)C)n2)=O)CN(C(C2(C(N)=O)CC2)=O)CCO1 c1(C(N2CC(CC)C(NC(c3nocc3Cl)=O)CC2)=O)c(C)ccc2nonc12 N1(C(c2cn(CCC)nc2)=O)CCC(C)C1CNC(=O)C(F)=C(C)C1CC1 N1(C(c2[nH]c(C)c(C)c2C)=O)CCC2(CC(NC(=O)CSC(F)F)CO2)C1 CCC(CC)CCCC(=O)N(CC#CC(=O)NC(C)C(C)C)C CC1CC(NC(=O)C2=CCSC2)CN1C(C1C2CN(C)CC12)=O C(CC(C(=O)NC(C)C(C)(C)C)NC(=O)Cn1nc(C)cc1C)=CC O=C(O)CC1CN(Sc2nccn2-c2ccccc2)c2ccc(Br)cc21 C1(C(N2CC(CCCNC(c3scc(C)n3)=O)OCC2)=O)CN2CCN1CC2C C1(CNC(c2cc(CCCC)oc2C)=O)CC(C)(C)CN1c1cnc(C#N)cn1 N1(C(CCC=C)=O)CCN(C(=O)CCCc2ccc(OC)cc2)CC1CCC C1(C(=O)OC(CC2(CNC(=O)OC(C)(C)C)CCCC2)=O)CCN(C)CC1(C)C N1(CCNC(=O)CCC2OCCO2)CCN(C(c2cscn2)=O)CC12CCC2 C(=O)(C(O)C(F)(F)F)N(C1(C(N2CCC(C(C)(C)O)CC2)=O)CC1)C C(CC(C)C(=O)N1CCN(C(=O)CNC(C2CSCC(=O)N2)=O)CC1)OC C1(C(=O)NCC2CCN(C(C(c3cccc(Cl)c3)CC)=O)C2)CC12CC(C)(C)C2 CS(=O)CCC(=O)N1CCC(NC(C2CCN(CC(F)(F)F)C2)=O)CC1 C12(C(=O)NCC(C)C#N)C(NC(c3cccc(C#N)c3)=O)C3CC1C2C3 C1(OO)(NC2CCC2)CCN(C(=O)COCC)C1.C(=O)(CNC(=O)CO)N(CC=C)C C12(CCNC(c3c(CC)ncnc3)=O)CCC(C1)N(C(=O)C(C)NC(C)=O)C2 C12(C(=O)Nc3cc(CC)cc(F)c3)CCN(C(C3(CC)CCCO3)=O)CCC1C2 C(=O)(C(CO)C(C)C)NC(CC)CNC(c1cn(C)nn1)=O CSC1=C(C(=O)NC2CC(O)CN(C(c3ccsc3)=O)C2)CCCC1 C(=O)(C(F)C(C)C(F)(F)F)NC12CC(Nc3ccc(C=CC(=O)OCC)o3)(C1)C2 C1(C(=O)NC2CC(NC(c3csc([N+](=O)[O-])c3)=O)C2)Cc2nncn2C1 C12(CNC(CC(=O)NCC3CC3)=O)CCC(C1)N(C(c1cnc(O)cc1O)=O)C2 N1(C(C(C(C)(C)C)OC)=O)CC2CCN(C(=O)COc3cncc(Cl)n3)CC12 C#CCC(C(N)=O)NC(=O)C(C1CC1)N(C)C(c1cc(F)c[nH]1)=O c1(CC)ccc(C(=O)NCC(F)CNC(C2CC2c2cccc(F)c2)=O)cc1N c1(OCCCC)ccc(-c2nnc(N(C(C)(C)C)C)n2CCOC)cc1 N1(C(c2on(C)c(=O)c2)=O)CCCN(C(=O)CCCC(F)F)C(CO)C1 N1(C(C(C)NC(=O)NC2CC2)=O)CCOC2(CCN(C(=O)C(F)=CC3CC3)CC2)C1 C1(OC)CN(C(c2cccn(CC(=O)OC)c2=O)=O)CC2(CCC2)C1.C(C)=O N1(C(CC=C=C)=O)CCCCCC1CNC(=O)C(=O)NC(c1ccc(F)cc1F)C C(CC(C)C)(C=O)N(C(C(CCC(C)=O)C)=O)C.C(C)(C)N C(N=C(NC(c1cccs1)C)NC1CCC(C(N)=O)CC1)c1cc(OC)no1 C(C(C)(C(F)(F)F)N(C)C)NC(=O)NC(c1cccc(OC)n1)C(F)(F)F C1(C(=O)NC2(C#C)CCOC2)CCC(O)CN1C(c1cncs1)=O C1(C(N(CCC(C)O)C)=O)CC12CCN(C(C1CN(C)C(=O)N1)=O)CC2 C1(NC(c2ccc(C)cc2)=O)CC(C)CN(Cc2cccc(C)c2O)C1 c1(C(C(=O)N(C2CC(NC(=O)CC(C)F)C2)CC)(C)C)ccc(F)c(Cl)c1 C(=O)(CS(=O)(=O)C1CCCC1)N(C1CN(C(C2(F)CCCOC2)=O)CCC1O)C N1(C(c2cnc(O)[nH]2)=O)CC2(CCCN2c2ncnc3c2CCC3)C1 CC1(C)COCCC1NC(=O)C(N1CCN(CC23COCC(CO2)C3)CC1)=O c1(CC(=O)CCCOCCNC(CC2C(OCC)CC2)=O)cc(C2CC2)no1 C1(C(N(CC(C)(C)O)CC)=O)CCC2CCC1N2C(C1CC2(CC2)CO1)=O c1(CCOCCOCCOC)ccc(C(=O)N)cc1C.C1(C)(C(=O)N)CC2CC2C1 CN1CCC(C)(CNC(=O)C(Cc2ccoc2)NC(=O)Cc2nc(=N)[nH][nH]2)C1 C(=O)(C(O)CC(F)(F)F)NCC(C(=O)NC1(C(COC)O)CC1)N(C)C CC(C)CC(CC(=O)N1CCOC(C2CC2)CC1)NC(=O)CSCCC1CC1 CCCCCC(CCCCCC)NC(c1cc(OC)ccn1)=O N1(C(C(C=C)(F)F)=O)CCC(C(=O)NOCC(=O)NC)CC12CCCC2 N1(C(c2c(C)nn[nH]2)=O)CCC(NC(c2cn3cccnc3n2)=O)C(CO)CC1 N1(C(c2cnc(C(N)=O)c(Cl)c2)=O)CCC2CN(C(C3CCCS3)=O)C2C1 c1(N(C(CCCc2cc(C)sc2C)=O)C)cccc2ncccc12 C(C(C(=O)NCCN(C)C1CC1)C(C)(C)C)NC(C(CCC)OC)=O C1(C(N2CCC2CNC(C2(N3CCC3)CCOCC2)=O)=O)CCC2(CC1)CC2 C1(C(N2CC(C(=O)N(C)CCN(C)C(C)=O)(CC)C2)=O)CCCC(=O)C1 c1(C(=O)NC(CNC(c2cc(OCC)no2)=O)(C)CO)ccc2nsnc2c1 N1(C(CCNC(=O)NC)=O)CCCCC(NC(=O)C(C)(O)C2CCC2)C1 N1(C(C2(C#N)CCCC2)=O)CC2(CCC2)CC1CNC(c1ccc(O)cc1)=O c1(C(N2C3(CN(C(Cc4c(C)cccc4)=O)C3)CC2)=O)ccc(S(C)(=O)=O)cc1 N1(C(CNC(=O)OCC2CCCC2)=O)CCC(F)(F)C(F)C1 c1(C(=O)NCC(CNC(C2CC(=O)N(O)C2)=O)OC)cc(Cl)n(C)n1 CC(C)C(C#N)C(=O)NC(C1CCCCC1)CNC(c1cncn(C)c1=O)=O c1(C(=O)NC(CC)CO)ccc(CNC(=O)Cc2cnsc2)o1 N1(C(C(C)=CC)=O)C2CCC1CC(NC(C1CCC1C(C)(C)C)=O)C2 C(=O)(CCCCCNC(N)=O)N1CCC(N(C(C=CC)=O)CC)CC1 C(=O)(C(C(C)(C)C)NC(=O)CCP(C)(C)=O)N(CC=C)CCO N1(C(=O)NCC(c2ccc(Br)cc2)C)CCOC(C(F)(F)F)C1 N1(C(=O)OC(C)(C)C)CC=C(C(=O)NC2CN(C(=O)C(N)=O)CC2(C)C)C1 C1(NC(C(CC=C)NC(C)=O)=O)C2CCC1N(C(=O)CCCCCC)C2 c1(OC)ccc(C)c(C(N2CCCC2CN(C)C(c2cocc2Br)=O)=O)n1 CC1CN(C(=O)CSc2cccs2)CC(C)C1NC(C1(O)CCCCC1)=O c1(CN2CCC3(C(C(=O)NC(CC(=O)OC)C)C3)C2)cccc2[nH]ccc12 C1(C(C)(C)CNC(=O)C=CBr)CCCCCN1C(=O)C(O)Cc1ccccc1 c1(CC)cc(Cl)ccc1C(=O)NCCc1cn(CCOC2CCOC2)nn1 c1(OC)ccc(C(N2CCC(NC(c3cncn(C)c3=O)=O)C2(C)C)=O)cc1C c1(NC2CCCC(N(C)C)C2)ccc(Br)c(S(=O)(=O)NCC(O)C2CC2)n1 c1(OCC)ccc2cc(C(N3CC(O)(CNC(=O)C(C)C(C)(F)F)C3)=O)[nH]c2c1 N1(C(c2ccc(C)o2)=O)CCC2C1CCCN2C(c1cncnc1C)=O CCC(CCC(=O)N1CCC(CO)C(O)C1)NC(=O)CCc1cccnc1 CN1CCC(C)(C(N2CCC(C)(C(=O)NCC3COCCOC3)C2)=O)C1 C(=O)(C1=CS(=O)CCC1)N1CCC(N(C(C(OC)C2CC2)=O)CC2CCCO2)CC1 c1(CC(C(=O)NC(C)CNC(c2ccc(Br)s2)=O)C)cccc(Cl)c1 c1(C(N2CCCN(C(C=C(CCC)C)=O)C(CO)C2)=O)cc(S(N)(=O)=O)c(C)o1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1C(=O)NC1CCCCC1)C(C)(C)C CN=S(C)(=O)c1ccc(C(=O)NC2CC(NC(=O)CCC(=O)NC(C)C)C2)cc1 C(=O)(C1CCCc2c[nH]nc21)N1C(CNC(CC(C)N(C)C)=O)CC2(CC2)C1 CCC(C(=O)NC12CCOC(CNC(c3ccnc(OC)c3)=O)(C1)C2)C(C)O c1(CC(N2CC(NC(c3ccc(CC)s3)=O)C(O)C2)=O)c[nH]c2ncccc12 C1(C(=O)NCC2C(C)CC2)(CNC(c2csc(Cl)n2)=O)CC(C)(C)C1 CN=c1nc(N2CCCC(C(=O)NC)C2)[nH]c(=NC(C)CCn2cc(C)cn2)[nH]1 C12(NC(c3n(CC)c(O)nc3)=O)CCCC1N(C(c1sc(C)cc1OC)=O)CC2 C(=O)(CS(=O)(=O)C1CCCC1)NCCCCN(C(=O)CCCCN(C)C)C(C)C C(C(C(=O)NC(CO)CCF)NC(=O)CCCC1CC1)SCC C(CC(CC)C(=O)NC1CC(C(=O)NOCc2ncccc2C)(SC)C1)=CC N1(C(c2n(C)nnc2)=O)CCC(C)(CNC(=O)CCNC(c2ccncc2)=O)C1 Cc1ccncc1Nc1ccc(Cc2cccc(NC=O)c2)cc1 CC1CCC(NC(c2cccc(N)c2)=O)CN1C(=O)C1=CCCCC1 Cc1nc(CC(=O)NC2(CNC(c3ccc(C(N)=O)[nH]3)=O)CC2)cs1 c1(C(c2n(CC=C)nnn2)(C)NCc2ocnc2C)ccc(C(Cl)Cl)cc1 C=CC(C)(CCOC)C(=O)N(CC(CC)NC(=O)CCc1cncc(F)c1)CC N1(C(c2ccc(C(C)=O)[nH]2)=O)CCC(C)CC1C(=O)NC1CN(S(C)(=O)=O)C1 CC(C)CC(F)(F)C(=O)NCC1COC(CNC(c2cccc(F)c2N)=O)C1 C(=O)(C(C(C)(C)C)SC)N(C1CCC(NC(C2C(=C)CC2)=O)CC1)C C1(NC(c2n(CC)ccc2)=O)CCC(CC(=O)NCc2cc(C#N)cs2)CC1 CC1(CNC(=O)CC2CC3CCC2C3)CCCN(C(=O)CCC2CC(F)(F)C2)C1 c1(C(=O)NCC2(C)N(C(C)(C)C)CCC2)ncc(N)cc1Cl C1(C)(CC(N2C(CCNC(C(C)c3ccco3)=O)CCC2)=O)CC(F)(F)C1 CCCC(CCC)=CC(=O)NC(c1cccc(CC)c1)CNC(C1(SC)CC1)=O Cc1cccc(CN(C(c2nonc2C)C(=O)NCc2n[nH]c(C)n2)C)c1 N1(C(C2C3CN(C(C(C)OC)=O)C2C3)=O)CC(=O)NCC1C(N)=O C(=O)(C(F)(F)CC(=O)NCCC1(CNC(c2cocc2C)=O)CC1)OC c1(OC)cc2c(cc1C(=O)NC1CCCC1NC(c1cccc[n+]1[O-])=O)CCC2 c12ccsc1NC2=O.C1(C(=O)OC)CCCN1C(=O)C(O)c1ccsc1 Cc1c(Cl)cnc(NC2CC3CCC2N(C(=O)CC2COCCO2)C3)c1C#N N1(C(c2cc(CO)on2)=O)CCCC2CCN(C(C3(CO)CC(F)(F)C3)=O)CC12 c1(C(C(=O)NC(C(C)NC(C(C)OC)=O)C)(F)F)ccc(C)cc1 C(C(=O)NC1CCOCC1)(C1=CCCCC1)N1C(C)COCC1 CCC(CC(=O)N1CCC1(C)CC(N1CCCCC1C(F)F)=O)CC(C)C c1(C(=O)OCC(COC(C)C)(C)C)ccc(Cl)c(F)c1.C(=O)CCCn1ccnn1 Cc1c(C(N2CC3CC2C3CNC(C2CCCC2C(C)C)=O)=O)noc1C1CC1 N1(C(C2CCC(=C)CC2)=O)CC(NC(c2cc(CCC)nc(O)c2)=O)C2(CC2)C1 CCC1=C(C(=O)NC2CC(C(=O)NCC3(CN=[N+]=[N-])CC3)C2(C)C)CCCO1 c1(SC)cc(C(=O)NC23COC(CNC(C4(C#N)CC4(C)C)=O)(C2)C3)ccn1 C1(CNC(C(CC)SC)=O)(COC)CCCN1C(=O)CCF C1(CC)CN(C(=NCCC)NCCN(S(=O)(=O)CC)CC)CC(C)S1 CC1=C(F)CN(C(=O)C(=O)NC2C3CCC(C3)C2c2ccccc2)CC1 C(CNC(C1CC1C(F)F)=O)(CC(F)(F)F)NC(c1c(=N)[nH]cnc1)=O CC(=O)CCCC(=O)NCC1CN(Cc2nc(C(C)C)no2)CCCO1 C1(C(=O)NCCN(C(=O)C(=Cc2cccnc2)F)CC)CCC(=O)N(C)C1 C1(C(N2CC(C#C)OCC2)=O)CC2CN(C(=O)CCCOC)CC2C1 CC1(C)CC(C(N2C3CCC2CN(C(C2(F)CCCCC2)=O)C3)=O)C(C)(C)O1 C1(CC(=O)NC2CC(NC(C3CCCO3)=O)C2)CCC=CCC1 C12(OCC)CCC(C(=O)NC(C)(CNC(c3occc3Cl)=O)C3CC3)(CC1)C2 N1(C(=O)Nc2c(CC)c(Cl)ccc2)CC(CO)OC2(CCC2)C1 N1(C(Cn2ncc(CC)c2)=O)CC(CNC(=O)C=C(C)C)C2(CCC2)C1 c1(C(=O)NCCC2CC(NC(c3c(C)ncnc3)=O)C2)csc2cncn12 C1(NC(C2CCC(C)O2)=O)(CF)CCN(C(=O)Cn2ccccc2=O)C1 C1(N(C(C2CC(C)(C(=O)OC)C2)=O)C)CCCN(C(=O)C(C)(C)NC(C)=O)C1 c1(C(N(CC(CC)NC(=O)Cc2ccc(Cl)cc2Cl)C)=O)ccc(F)c(C)c1 Cc1cc(C(=O)NCC2CCN2C(=O)C=Cc2cscn2)cc([N+](=O)[O-])c1O Cc1cccc2[nH]cc(C(=O)NCC3CN(C(C4CC=CC4)=O)CC3(C)C)c12 C(CCCCCC(=O)NCCCc1nccs1)NC(c1cccc(C#N)c1)=O c1(C(N2C3C(NC(c4ccn(C)n4)=O)CC(CC3)C2)=O)ccc2c(c1)COCO2 N1(C(C2CCN(C)C2)=O)CCCC12CCCN(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 C1(CNC(C=C=C(C)C)=O)CC(F)(F)CN1C(=O)C(=O)NCC1CC1 C1(C(=O)NCC2(NC(=O)CC3CCC(O)CC3)CC2)CCC2(CC1)CC2 C=C(C)C(CC(=O)NCC1CCN(C(c2cc(CC)nn2C)=O)C(C)C1)OCC N1(C(C(C)SC)=O)CCCC2(CCCN2C(=O)CC2CC2(Cl)Cl)C1 C1(CNC(C2(C)CC=CC2)=O)COCCN(CCCCCO)C1 C1(C(N2CC(C)(O)C2)=O)(COC)C=CCN1C(c1cc(OC)nn1C)=O Cc1cc(Cl)nc(Cl)c1C(N1CCOC(CNS(=O)(=O)CC#N)C1)=O CCC(CCC(=O)NCCC(C)(C)CO)NC(C1CC(C(C)C)C1)=O c1(C(=O)NC2(C3CC3)CCN(C(=O)CCCC3CC3)C2)ccc2c(c1)COCC2 N1(CCC(=O)NCCCN(C(=O)COC2CCOC2)CC)CCCS1(=O)=O N1(C(C2C(C)CNCC2)=O)CCC(O)CC1C(N1CCOC(C)(C)C1)=O Cc1cc2c(CC(=O)NCC(C)NC(c3snnc3C3CC3)=O)csc2s1 N1(C(C(Cn2ccc(C)n2)C)=O)CC2CC1CN(C(c1cc(N)cnc1C)=O)C2 C1(SC(C)(C)C)CC2CC(C1)N(C(=O)N(C1(C)CCCC1)C(c1c(C)scc1)=O)C2 C=Cn1nncc1C(=O)N(C)CCNC(=O)CCc1ccc(OC(F)(F)F)cc1 C1(NC(CCC#C)=O)CN(C(=O)C(O)(C2CC2)C2CC2)CCC1O C1(C)(C(=O)NCCCCC)CCCN(Cc2c(C)n[nH]c2C)C1 CCCC(C)C(=O)NCC(CC(=O)NCC(C)C(C)O)C1CCC1 N1(C(c2c(C)cn(C)n2)=O)CCCOC(CNC(c2cc(Cl)c[nH]2)=O)C1 c1(C(N(C)CC2(O)CN(C(C(C)(C)OCC)=O)C2)=O)cn2c(n1)C(C)CCC2 CC1(C)CCC(CNC(c2cc(Cl)c(Cl)[nH]2)=O)N(C(c2ccc(F)cc2F)=O)C1 c1(C(=O)NCCCN(C(C)C)C(c2cn(-c3ncccn3)cn2)=O)cccnc1 C(CCCCC(=O)N(CCC(C)C)C)OCc1cn(-c2ccc(C)o2)nn1 N1(C(C2ON=C(CC)C2)=O)CCCCC(C(=O)N(CC)CC2CCOCC2)C1 C=CC1(C(N2CC(C(C)(C)O)(CNC(=O)Cn3nccc3C)C2)=O)CCC1 N1(C(Cc2ccn(C(C)C)n2)=O)CC2(CCN(C(c3ccnnc3O)=O)CC2)C1 C1(C(N(C)CC2COCCN2C(=O)CC2CCOCC2)=O)CCc2n[nH]cc2C1 N1(C(C23C(NC(c4c(CC)cccc4)=O)C4CC2C3C4)=O)CCc2cccc(C)c21 C1(C(C)(C)C)CCN(C(c2ccco2)=O)C(CNC(c2cc(O)nc(Cl)c2)=O)C1 c1(CNC(CCCn2cc(-c3ccc(=N)[nH]c3)nn2)=O)ccc2nc(O)[nH]c2n1 C1(C(=O)NCCCCNC(C2CCC=CCC2)=O)CCc2nccn2CC1 c1(C(=O)NCCC2(C(N(C)CC3(C)CCCC3)=O)CCC2)sccc1C#N N1(C(C(=O)NC(C)C)=O)CCCC12CCCN(Cc1ccccc1)C2=O C1(CC(=O)NCC(COCC)C)CC(O)CN1C(c1cccc(C)c1)=O C1(NC(C2C(NC(CC3C(C)(C)C3)=O)CCOC2)=O)CN2CCCC1C2 N1(C(C2(CC)COC2)=O)CCN(C)C(C(=O)N(C2CCC(F)(F)C2)C)C1 C1(CCCC)CCCC1(c1nnnn1C1COC1)NC1(CC2CCC2)CC1 N1(C(c2ccc(CCC)s2)=O)CC2CCN(C(=O)CCN(CC)CC)C2C1 c1(OC)ccc(C(=O)NCC(CO)NC(=O)C(F)(F)C2(O)CCC2)nc1OC N1(C(COCCN(C(C(C2CC2)OC)=O)C)=O)CCCC(C2(C)CC2)C1 N1(CCOCCOCCCC)CC2C(C(=O)Nc3nnc(C)s3)C2C1 Cc1nc(C)c(CNC(C2(C3CCCN3C(=O)C(C)C3CCC3)CC2)=O)[nH]1 C(CCCCC(=O)N1CCOC(F)(F)C1)NC(CC(CC)O)=O C1(C(=O)NCC2CCN(C(C(COC(C)C)NC(C)=O)=O)C2)CCC(C)(C)CC1 c1(C(N(CCN(C(=O)CN2OC(C)(C)CC2=O)C)C)=O)cncc(Cl)c1Cl c1(CN(C(C)Cc2ccccc2F)C)nc2cc(F)c(F)cc2[nH]1 N1(C(C(C=C)C)=O)CCC2(CCN(C(c3ccc(OC)nc3)=O)C2)C1 N1(C(C2CCCC(C)C2)=O)CCCC(C)(C)C1CNC(C1C2CC3C(C2)C13)=O O=S(=O)(c1c(F)cc(F)cc1F)N1CCC(O)CC1C(N1CCCC(F)CC1)=O c1(CC(=O)N(CC)CC2CCCN2C(C2CNC(=O)N2)=O)c[nH]c2ccccc12 S(=O)(=O)(c1cnn(CCF)c1)NC(C1OCC(C)C1)(C)C C(N=c1[nH]c(C(=O)NCCOCC)cs1)c1ccc(C#C)s1 C(CC(=O)NC(c1cn[nH]c1)C)(C1CC1)NC(C1CC(C)C1)=O N1(c2nc(N3CCN(CC)CC3)c3c(n2)CCS3)CCc2c(C)cccc2C1 C1(NC(CN(C)C)=O)CCCC(C(=O)N(C23CC(C2)C3)CCO)CC1 c1(CNC(c2ccn(CCNC(c3cnc(Cl)s3)=O)c2)=O)ncccc1Cl c1(CNC(c2nc(-c3c(-c4ccc(C)o4)n[nH]c3)sc2)=O)cccn(C)c1=O CC1CN2CCN1C(C(=O)NC1CN(C(c3ccc4nn[nH]c4n3)=O)CC1F)C2 c1(C(=O)NC2(CN(C)C(C3CC(O)C(F)C3)=O)CC2)cc(Br)cnc1N C=C=CC(C)C(=O)NC(Cn1cccn1)C(=O)NC1C(=O)NCC1CO CCCCC(F)C(=O)NCC(C(=O)N(CCOC)CC1CC1)OC C1(O)(CNC(c2cc(F)cc(F)c2)(CC)C)CCCN(Cc2ccccc2)C1 Cc1c(C(=O)N(CC(C)NC(C2CC2c2ccc(F)cn2)=O)C)sc2nccn12 Cc1ccc(F)c(OCC(=O)N(C2CCCN(C(C3CCCCO3)=O)CC2)C)c1 c1(OC(C(=O)NCC(C)NC(c2nc(CC)oc2C)=O)C)cc(Cl)ccc1Cl c1(C(=O)NC2(C(N3CCC(CC)CC3)=O)CC2(C)C)ncc(C)cc1F Cc1cnc(C(N2CC(C)C(C)(CNC(=O)CS(N)(=O)=O)C2)=O)cc1C c1(OC)ccc2[nH]c(C(=O)NC(C)CNC(C3(C)CCCC3(F)F)=O)cc2c1Cl C(C(=O)NNc1ncnc(C)c1)C1NC(C(=O)OC)C(F)(F)CC1 N1(C(Cc2ccc(SC)cc2)=O)CC(NC(=O)C(C)S(C)(=O)=O)CC(F)C1 N1(C2CC(N)C2)CCC(CN(C)C(N2CCOCC2)=O)CC1 c1(C(=O)NCC(=O)NCC(N2CC(OC(=O)NC)C2)=O)cc(C)co1 C1(NC(=O)NCC(C2CCOCC2)F)CN2CCC1C2 Cc1c(C(=O)NCCC2CN(C(C3CC(F)C3)=O)CCO2)ccn1C1CC1 N1(C(c2c(C(C)C)con2)=O)CCN(C(=O)CCCSC(C)(C)C)CC12CC2 c1(C(C)C(=O)C2C3C(CC2)NCCC2CSCCN2C3=O)ccc(F)cc1F n1(CC(=O)NCCN(CCC)C(C2CCC2(OC)OC)=O)cccnc1=O N1(C(Cc2n(C)ccn2)=O)CCC(CO)(NC(=O)CSc2nnnn2C)CC1 N1(C(C(N2CCSCC2)C)=O)CC(NC(=O)Cc2nc(=N)[nH][nH]2)CC12CCOC2 CCC(N=c1[nH]c(=NC2CCSC2)[nH]c2c1CCCCC2)c1cccc(OC)n1 c1(C(N(C2CCCC2)CC#CC)=O)ncoc1CNC(=O)CC1(C)CC1 C12(C(N(CC(C)CNC(C3CC3OC(C)(C)C)=O)C)=O)CCC(CO1)C2 CC1CCN(C(=O)C(=O)Nc2ccc(Cl)cc2)CC1N(C(=O)CCC(C)(C)F)C c1(OCCC(=O)NC2CCC(CNC(c3ccc(F)o3)=O)C2)cccnc1 N1(C(C2CC(N(C)C)C2)=O)CCCC(F)(CNC(=O)CC2COCCO2)C1 C1(F)(CNC(C2CC3CCC2O3)=O)CCN(C(=O)C=Cc2ncc[nH]2)C1 c1(OC)cc2c(cc1C(=O)NCCC1CCN(Cc3cccs3)C1)OCO2 N1(C(=O)Cn2cccnc2=O)CCC2OCCN(C(c3ccoc3Cl)=O)C2C1 c1(OC(C)C(=O)NCC2COCCN2C(C2CC=CCC2)=O)ccc(F)cc1Cl C1(C(N)=O)CCCN(CCC(=O)C2CC2)C1.C1(C(=O)NC2(CN)CCC2)CC(F)(CO)C1 C(CC(C(C)C)NC(=O)CSCCC(F)(F)F)NC(C1C(C)=C1)=O CC(C(=O)NCCCNC(=O)CNc1ccc(C(F)(F)F)cn1)C(F)F C(C(=O)NC1CN(C(C2(C)CCCO2)=O)C1)(C(C)C)NC(=O)OC C(C(=O)NCC#CCNC(c1ccnnc1O)=O)(C(C)C)c1cnc(C)s1 C(C)(C)(C(=O)NCC(CC)NC(=O)CC1CC1COc1ccccc1)OCC FC1(F)CC2CC1CC2(c1nnnn1CC1CC1)NCc1nnc(C2CC2)o1 C1(O)(CC(N2CCC(CC3N(C(CCC=C)=O)CCC3)CC2)=O)CCCN(C)C1 C1(C(=O)NCCC(=O)NC)CCN(c2ncc(Cc3ccccc3)cn2)CC1 N(C(=NCC1CCC1)NCc1ccnn1C)C(c1cncs1)C C12(C(N3C(C)CCC(NC(c4n(CCC)ncc4)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 c1(-c2n(C(C3(C)CC3)C)nc(-c3nccs3)n2)c[nH]c2cc(C)ccc2c1=O C1(C(=O)NC2C(NC(Cc3nnn(C(C)(C)C)n3)=O)C2)CCCN(C2CC2)C1 C1(C(C)NC(c2cnns2)=O)CN(C(=O)Cc2sc(O)nc2O)CCO1 c1(CSCC)ccc(Cl)c(C(=O)NCC2COCC2NC(=O)CC2(C)CCC2)c1 CCCCCC(=O)NC(c1ccccc1F)CNC(c1onc(C)c1C(F)F)=O C1(C(=O)NC(C2CCCO2)CO)(COC)CN(C(=O)C=CCO)C1 C=CC1CCCN(C(c2cncc(C(=O)NC(C)C)c2)=O)C1.C12(CC1)C(=O)N2 N1(C(C(CCC)C#N)=O)CCC(C)(C)C(NC(=O)C(C)OC2CCCC2)C1 N1(C(C(CC2CC2)OC)=O)CCCC(CNC(=O)COC2CC2)CC1 C1(N(C(Cc2c(C)n[nH]c2C)=O)C)CCN(C(C2OCCC2C(C)C)=O)CC1C Cc1cc(C)c(C#N)c(NCCC2CCC(NC(=O)CCc3nc[nH]n3)C2)n1 N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)COc2ccccc2Cl)C(CF)C1 C(C(O)CCNC(C1CCCC1)=O)NC(c1cnnn1-c1ccccc1)=O C1(O)(CNC(CN(CC)CC)=O)CCN(C(C2(C#N)CCC2)=O)C1 C1(CN(OC)C2CCC2)CC2C=CC1N(C(C1(OCC)CCOCC1)=O)C2 C1(OCC)CCCN(N2CCN(c3ccc4oc(O)nc4c3)CC2)C1C C(=O)(C#CC1CCCCO1)NCC(CNC(C1CC(C#C)(O)C1)=O)C c1(C(N2CC(CNC(c3cnco3)=O)C(C(F)(F)F)C2)=O)cnc2n1CCS2 c1(CC)oc(C)cc1C(=O)NC(C)CCNC(=O)C(C)(CO)OC c1(NC(C(C)OC(=O)Cn2c(O)nnc2O)=O)cc(F)cc(F)c1 N1(C(Cc2ccc(C)s2)=O)CCC(NC(=O)CC2CC3(CC3)C2)CC1C1CC1 C1(NC(c2c(C)cno2)=O)CCCC1(C)CN(C)C(C1CC12CCCC2)=O Cc1ccc(N2CCCC(CNC(C3CCCC3C)=O)C2)c([N+](=O)[O-])c1 N1(C(CCCN(C(=O)OC)C)=O)CCCC(C(N2CCC2CN(C)C)=O)CC1 S(=O)(=O)(c1ccc(Br)cc1NCC1(CN(C)C)CCOC1)NC1(COC)CCC1 N1(C(CCC(=C)Cl)=O)CC2(CC(C(=O)NOC(C)(C)CC3CC3)CO2)C1 C(=O)(C1OCCc2c(O)cccc21)N1CCCC(CN(C(=O)CSC2CC2)C)C1 NS(=O)(=O)CC(=O)NCC1CC(F)(CNC(=O)CSC(F)(F)F)C1 C(=O)(CCCCC#Cc1ccccc1)N1CCN(C(C(CC)OC)=O)CC1CF C1(NC(C(C)CO)=O)CC2CCCC(C1)N2C(=O)CS(=O)(=O)NC1CC1 c1(C(=O)NC2CN(C(=O)C3=COCC3)CC23CC3)cc(Cl)c(Cl)cc1O Cn1c(C(N2CCN(C(C3CCCCCS3)=O)CC2CCO)=O)cnc1[N+](=O)[O-] c1(C(C)N(C(=O)C(=O)NCC(N)CO)C)nc(-c2ccccc2)cs1 N1(C(C2C(=C)C2)=O)CC2COCC2(C(=O)NC23CCCC2C3)C1 N1(C(c2n(C)nnc2)=O)CCN(C2CCN(C(=O)COC3CCC3)C2)CC1 c1(SC)cc(F)ccc1C(N1CC(N(C(=O)CNC(=O)CN(C)C)C)C1)=O c1(C(C)F)ccc(C(=O)N(C)CCN(C)C(c2ncoc2Br)=O)cc1 C(=O)(CCC(C)NC(C12CC1CN(C(c1cnc(O)o1)=O)C2)=O)OC C1(C(=O)NCCCCCC2CC2)(NC(C=NOC)=O)CCCC1C c1(OC)cccc(C(O)C(C2CC2)NC(=O)NC2CCC(CCO)CC2)c1 c1(CNC(=O)NCC23CCCC2(O)C(=O)N3)cc(F)cc2ccncc12 c1(-c2n(CCOC)nc(COC)n2)nccc(OC(C)C)c1Br N1(C(CCC=C)=O)CC2CC1CN2C(C1CCCC(F)(F)C1)=O C1(C(=O)NCC(C(CC)C)N)CC2C=CC1NC2 c1(C(=O)NC2CCN(C(CC3CCCC(OC)C3)=O)CC2)ccc2nc[nH]c2c1 N1(C(C2CN(CC)C(=O)CC2)=O)CC(CO)C2(C1)CN(C(=O)Cn1cccn1)C2 c12nnc(n1CC(C)C)CC1CCN2C1.C(C)(C(C)C)OCCOC C12(NC(Cc3n(C)nc(C(F)(F)F)c3)=O)CCC(CC1n1cc(CO)nn1)C2 C(=O)(C(C)(O)C1CC1)NC(n1cc(COC(=N)O)nn1)C Cc1cc(C(=O)NC2CN(C(C3COCCOC3)=O)CC2C)ccn1 c1(N2CC3C(CNC(CC(=O)OCC)=O)C3C2)nc(CC)nc(C)c1C(=O)OC C1(NC(=O)CCCF)CCCCC12CCN(C(=O)Cc1cc(F)cc(F)c1)C2 c1(C2C(C(=O)NC(C)CCCO)CC2)cccc(F)c1 C(C(=O)NCC(C)(C)CNC(C1(CO)CCC1)=O)(C(C)C)NC(CC(C)C)=O c1(C(N(CC(C)N(C(Cc2cc(C)no2)=O)C)C)=O)coc2c1CS(=O)(=O)C2 c1(OC(C)C(=O)NCC2(CNC(C3CCCCS3)=O)CCC2)ccccc1C#N Cc1cnc(NCCc2c(Cl)cccc2Cl)c(S(=O)(=O)NC2CC3CCC2C3)c1 CCC(C)(F)C(=O)NCC(c1cccc(OC)c1)NC(c1nccnc1C)=O c1(C(C)(C)C)nccc(C(=O)NC2CC(CNC(C3(O)COC3)=O)C2)n1 C#CC(CCC)NC(=O)C(C)(C)NC(=O)C(C)COC(C)=O CN=S(C)(=O)c1ccc(C(=O)NC(C)CNC(c2cc(F)ccc2O)=O)cc1 Cc1c(F)ccc(Cl)c1C(N1CC2CCC2(CNC(c2cc(Cl)cn2C)=O)C1)=O c1(CCC(=O)NCC(C)(C2CC2)NC(C(C)(C)OCC)=O)n[nH]c2c1CCCC2 C1(NC(c2cn(CC(C)C)nc2)=O)CCN(C(=O)Cc2cscn2)CCC1CO Cc1cc(C(=O)NCC2CC2NC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)c(F)cc1N n1(CCOC)cc(C(=O)NC(C)CC(C)NC(c2cc(C)ns2)=O)c(C)n1 c1(C(=O)NCC2N(C(CS(CC)=O)=O)CCC2)cc(F)cc(S(N)(=O)=O)c1 c1(C(=O)NC2CC(NC(CC(CCC)C)=O)C2)c(Br)ccc(F)c1OC C1(NC(c2n(C)c(S)nn2)=O)CCC2CC1CN2C(c1n[nH]cc1F)=O N1(C(C23CCC(OC)C2C3)=O)C(C(N2CC=CCC2)=O)CCC12CC2 c1(CC)c(C(=O)N(C2CCC(NC(=O)CC3(CSC)CC3)CC2)C)csc1C C1(NC(CCC(=O)NCC)=O)CCN(C(=O)C(F)C(C)(C)O)C12CC2 C12(CC(=O)NC3CC3CNC(=O)COc3cccnc3)CCCC1C2 c1(NC)cncc(C(=O)NC(C(N2CCC(C(C)C#N)CC2)=O)C2CCCO2)c1 Cc1ccccc1-c1nc(C2CCN(C)C2=O)n(-c2ccn(C)n2)n1 c1(C(=O)O)ccc(F)c(CN2CCC3(CC3C(N3CCC(F)C(O)C3)=O)C2)c1 C1(CN(C(Cc2ncc(C)o2)=O)C)CCN(C(=O)CSc2cccc[n+]2[O-])CC1 Cc1nc(C)c(C(=O)NC2CN(C(=O)C=CSCc3ccco3)C3CC23)[nH]1 N1(C(c2ccc(COC)o2)=O)CC2(C1)CN(C(=O)C(C)SCC)CC2CO CCCCCC(C)C(=O)N1C(C(=O)Nc2ccc(F)cc2Cl)COCC1 c1(C(N(CCC=C)CCOC)=O)cn2ccc(-c3cc4sccc4s3)cc2n1 N1(C(C(C)(C)F)=O)CCN(C(c2cc(F)ccc2Br)=O)C(CO)C1 Cc1csc2c(N3CCC(C)(C(=O)NCC(C)O)C3)ncnc12 N1(C(COCCCCC)=O)CC(NC(=O)CC2CC23CC3)C(n2ccnn2)C1 C1(COC2CCN(c3n(C)nnn3)CC2)CC2CCC1C2.c1ccc(Br)cc1.O1NC1=O Nc1ncc(C(=O)NCC2CC(C(=O)NCC3(CO)CCC3)C2)cc1CO c1(C(N(C(C(=O)NCC=CCOC)C)C)=O)ccsc1C#N C12(NC(C=C(C)C(F)F)=O)CCC(CC1)N(C(=O)Cc1cn(C)nc1C)C2 N1(C(C2(CSC)CCC2)=O)CCCC(C(=O)NC2COCCC2OC)C1 c1(NC(N2CC(CO)CC(NC(N3CCS(=O)CC3)=O)C2)=O)cccc([N+](=O)[O-])c1 C=C(C)CC(C(=O)NCCC1(C)CCOCC1)NC(=O)CC1CCCO1 C1(O)CCCCC1(F)F.N1(C(C)=O)CCC(CC(=O)NOCCCC2CC2)CC1 C(=O)(C1CCCc2nn[nH]c21)C(C)C.C1(C(NCCNC)=O)CCN(C)C(=O)C1 CCCCCC(O)CC(=O)N1CCC(NC(C2CCC(CC)CC2)=O)C(O)C1 c1(C(N(C2CN(C(c3c(C)nc(CCC)o3)=O)C2)C)=O)cnc2ccccc2c1 C1(C(=O)Nc2ncn(C)c2)CCCN(C(C2CC3CC3C2)=O)CC1 CCS(=O)CC(=O)NC1CC(CNC(=O)Cc2ccccc2C)C1 C1(C(C)NC(C(C)OCCC=C)=O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1 c1(C(N2C(C(=O)NCCC=C)C(C)C2)=O)c(F)cc(Br)cc1F C(CC(C)(C)C)(C(=O)NCCNC(=O)C(C)Cn1ccc(C)n1)OC c1(CN2CCC(CNC(c3ncc(C)nc3)=O)C2)cc(F)cc([N+](=O)[O-])c1 C1(CC)OCCC1C(=O)NCC12CC(NC(c3c[nH]nc3C)=O)(C1)C2 CC(C)(C)C(CNC(c1c[nH]c(=N)s1)=O)NC(c1cn(-c2ccccc2)cn1)=O c1(C(C)C(=O)NC2CC(COC(F)(F)F)C2)ccc(Br)cc1 c1(C(N)=O)ccnc(N(C2CCC(N(C)C)C2)C2CC2)n1 C=C=C(C)CC(=O)NCCCNC(=O)C(O)Cc1cccc(C(F)(F)F)c1 C1(C#N)(C(=O)NCCC(C)NC(C2N(C(C)=O)CS(=O)(=O)C2)=O)CCCCCC1 CC1(C)C(CNC(c2cnc(=N)[nH]c2)=O)CCN1C(c1coc(Br)n1)=O CC1CCc2nc(CNC(=O)C(=O)N(C)C(c3ccccn3)C)sc2C1 N1(C(Cc2cccc(OCC)c2)=O)CCOCC(F)(CNC(=O)C(C)C(C)C)C1 c1(OC)ccc(CC(=O)NCCSc2ccccc2C)cc1 C1(NC(CSCC=C)=O)CN(C(=O)CC2(C)CCOC2)CC1OC c1(C(C)(C)C)cc(C(=O)NCC2CCCN2C(=O)C(C#N)=CC(N)=O)no1 Cc1ccc2c(c1)C=C(C(=O)NCC=CCNC(c1ccnnc1S)=O)CO2 N1(C(c2cnc(-c3ccccc3)nc2)=O)CC2(CC(C3CC3)=NO2)C1 c1(CN(C(c2ccc(COC)cc2)C(=O)NC(CC)(C)C)C)c(C)cccc1C C(CC(=O)N(C)CC1CCN(C(c2ccc(Br)o2)=O)C1)(C(C)C)OCC c1(C(=O)NC(C)CCCNC(c2ccoc2C(F)(F)F)=O)nccnc1N c1(CC)ccc(C(N2CCC2CNC(=O)CCc2cc(C)nn2C)=O)c(C)n1 C1(NC(c2c(SC)cc(F)cc2)=O)COC2(CCCN(C(=O)COC3CC3)C2)C1 N(C(=NCCCN1CCCCC1)NCc1ccccc1)Cc1cnn(CC)n1 N1(C(=O)OC(C)(C)C)CC(CNC2CC3CC2C3)OCC1(C)C C1(COCC)CC2CCC1N2C(=O)CCC1(C)CC1.C12CCCN1C2=O CC1=CCN(C(=O)C(C)(C)C2CCCN2C(=O)COC2C=CCC2)C1 n1(CC(=O)N(CCO)Cc2nc(C)[nH]n2)c2ccccc2c(=O)c2ccccc12 C1(CC(=O)NC2(CC)CCC2)CCN(C(=O)C=C(C)C2CC2)C(C(N)=O)C1 N1(C(C(CCCC)NC(=O)CN2CCCCC2)=O)CC2CCC(C1)C(=O)O2 CC1(C)CCC(C(=O)NCCN(C2CCCC2)C(C2CCCS2)=O)OC1 C1(C(N2CCCC(COC)C2)=O)C2CC(CC2F)N1C(=O)C(C)S c1(OC)cc(N2CC=CC(NC(c3cnc(F)c(C)c3)=O)C2)nc(OC)n1 CC1CC(NC(CNC(c2ncoc2CCC(F)(F)F)=O)=O)CN1C(=O)CCF C(=O)(CC(CNC(c1ccc(Cl)cn1)=O)C1CCC1)N(C1(CO)CCCC1)C N1(C(CC2C(C)(C)OCC2)=O)CCC2CC1CN2C(=O)CCc1ccncc1 C1(NC(c2ccc([N+](=O)[O-])s2)=O)CC12CCN(C(=O)CC1CSCCS1)CC2 C1(C(=O)NCCC(C(C)C)OC)CCC2(CC2)N1C(c1cc2n(n1)CCO2)=O Cc1nccnc1C(N1CC(OC2CCN(C(=O)CN3CCOCC3)CC2)C1)=O C(C(=O)NN1CCCC1C(N1CCOC(C2CC2)C1)=O)c1nc(C(C)C)oc1 CN1CCNC(=O)C12CC(N=c1[nH]c(N3CCSCC3)nc3ccsc13)C2 C(C(C(=O)NCCc1cccc(F)n1)C(C)C)NC(C1C(CC(C)C)C1)=O C1(O)(CNC(C2CCCCCC2)=O)CCN(C(c2ccc(CCF)cc2)=O)CC1 c1(C(=O)NC(C2CCN(C(C3(N(C)C)CC3)=O)C2)C)cn(C)ccc1=O c1(OC)cccc2c1C(C(=O)NC1CC1NC(c1cnc(C)cn1)=O)CC2 O=C(CCCC(F)(F)CO)NC1(CCN=c2ccnc[nH]2)CN(Cc2ccccc2)C1 c1(-n2c(C)ccn2)ccc(C(=O)NCC(CCl)NC(c2cc[n+]([O-])cc2)=O)cc1 CN1C(=O)CCC1C(=O)NC1CCC(NC(c2ccnn2C2CC2)=O)CC1 C=CC1(C(N2CCN(C(c3cc4ccsc4s3)=O)CC2CCO)=O)CCOCC1 c1(CS(=O)(=O)NCC2CCCN(C(c3cccc(OC)c3)=O)C2)cc(O)ccc1F Cc1nn2c(c1C(=O)NC(C1CCOC1)CNC(=O)CCCCC#N)CCCC2 c1(OC)nc(C(=O)N2CC(n3cc(C4CC(=O)NC4=O)nn3)CO2)cc(O)n1 c1(OC)cccc(Br)c1C(N1CCN(C(=O)C2=NOCC2)CC1CF)=O CCC(CNC(C1CCCCC1OC)=O)(CC)C(=O)Nc1cccc(F)c1 c1(CC(C)C)ccc(C(N2CC(NC(=O)CC3CCCCCC3)C2)=O)cc1 CC(C)CC(CNC(c1nncn1C1CC1)=O)NC(c1scnc1C(F)(F)F)=O c1(NCCOCC(=C)C)cc(Br)ccc1S(=O)(=O)NCCO c1(C(=O)NC2C(NC(C3CN(C)C3)=O)C2)cc2c(cn1)OCCO2 c1(SCCNC(c2ccsc2OC)c2n(CC)nnn2)cccc(C)c1 C=C(C)CCC(=O)NCC1(F)CC(NC(c2ccn(CC)c2C)=O)C1 Cc1cc(CCC(=O)NCCC2(CNc3ncncc3I)CC2)cc(C)c1 C1(NC(CCC#CC)=O)CC12CC(NC(C13CC(c4ccccc4)C1C3)=O)C2 C(CC(C)C)(C(=O)N1C2CCC(C2)C1CC(=O)NC1CC(O)C(F)C1)OC C(=O)(CCC(=O)c1ccccc1Br)NCCCN(C(=O)CCCN(C)C)C c1(CC)ccc(C(C)(C)C(=O)NCCC2(CNC(c3ccc(F)s3)=O)CC2)cc1 c1(C(=O)NCC2C(CNC(c3cc(C)nn3C3CCC3)=O)C2)cccc(O)c1Cl C1(NC(c2csc(C)c2C)=O)CC2(CCN(C(c3ncnc4ccsc34)=O)C2)C1 C(=O)(C1CCCc2ccccc21)NCC1CC(NC(C(CN(CC)CC)F)=O)C1 C1(C2(C(=O)OC)CC2)CCCN1C(C)=O.c1(C(C2CCCCC2)N)c[nH]cc1CN c1(C(=O)NC(CNC(C(=O)NCC)=O)(C)CC(C)C)ccc2c(c1)CCCC2=O n1(CC(=O)NC2CCCC(NC(C3(F)CC3)=O)CC2)cnc2sccc2c1=O C1(c2n(CCOC)nnn2)(NCc2cnn(-c3ccc(F)nc3)c2)CC(F)(F)C1 N1(C(c2cc(C(CC)CC)no2)=O)CC2CC(C1)C2NC(c1cnsc1)=O C1(C#N)(C(=O)OC(C)C(=O)NC(C2CCCC2)=O)CCN(C(=O)CC2CC2)CC1 C1(CNC(C=C(C)c2cccs2)=O)CN(C(=O)CC2CSCCS2)CC1(C)C C1(C(N(CC(CNC(CCc2scc(C)n2)=O)C)C)=O)CCc2c(ncn2C)C1 C1(CCN=C(NCc2nnc(C)s2)NCC2CCCO2)COc2ccccc2O1 C12(CC(=O)NCC(CO)NC(=O)C=Cc3nccs3)CCC(CC1)C2 c1(C(N(CCNC(CC2CC(CC)OCC2)=O)C)=O)cc(C#N)c2n1CCCC2 CCCCC(CNC(=O)Cn1ncn(C)c1=O)NC(c1scnc1C1CC1)=O C1(CNC(c2c(C)ccs2)=O)CC12CCN(C(=O)CCOC1CCC1)CC2 N1(C(COCCC)=O)CCC(OCCC2CCCCC2)C1 N1(C(C2CCCN(C(C)=O)C2)=O)CCCC(CNC(=O)CC2CCCCC2)CC1 C1(CC=C)(C(=O)NCCCCCN(C(=O)C=CCF)CC)CCOC1 C=C(C)C(CC(=O)NCC(C)(C(C)C)NC(=O)Cc1ccc(Cl)cc1)OCC C(c1nc(C)cs1)=CC(=O)N(C(CN(C(CNC(=O)OC)=O)C)C)C C(=O)(C(C)(C=C)CCOC)NCc1cc(C(N2CCC(C(=O)NC)C2C)=O)n(C)n1 CCC(CC)C(C)C(=O)NC1CN(C(C2(CSC)CC2)=O)CC1C C1(C)(CNC(C2CC(n3cc(CN(C)CCO)nn3)C2)=O)COCCO1 C1(CC(N2CCC(C)C2)=O)CCCCN1CC1CC1.Cc1nscc1-c1c[nH]nn1 c1(C(C)C)cc(C(=O)N(C)C)nc2ccccc12.c12cc-1ccc2O Cn1nc2c(c1NC(c1c(Cl)cc(Cl)nc1N)=O)COCC2 c1(C(=O)NC2CN(C(c3cccc(CC)c3F)=O)C2)cc2sc(N(C)C)nc2s1 CCC(C#N)C(=O)NCC(C)(C)NC(c1coc(-c2cccnc2)n1)=O CC1CCN(C(=O)CC2CCN(C)C2=O)CC1NC(C1CC(OC(C)(C)C)C1)=O c1(C(N2CCC(CCNC(CC(C=C)(C)O)=O)CC2)=O)ccc2ncc(C)n2c1 C(=O)(C1=CC(C)(C)C1)NCC(CC)NC(c1cnoc1-c1ccccc1)=O C1(C(N(CC(C)(C)CNC(=O)C(c2ccc(Cl)s2)C)CC)=O)NC(=O)OC1C C1(NC(C23C(C)OC(C)(C2)C3)=O)CCCC2CN(C(=O)CC3CCC(=O)N3)CC12 c1(C(=O)NCC2CC2CO)ccc(F)c(CNC(c2ccc(Br)cc2O)=O)c1 C(C(C)(CC)C(=O)N1CCC(N(C)C)C1)NC(c1n(CC)c(O)nc1)=O c1(NC(CCOC2CN(C(c3cc(CC)no3)=O)C2)=O)cnc(O)c(F)c1 c1(C(=O)NC(C2OCCN(C(c3c(CC)ccs3)=O)C2)C)cc(F)cc(C)c1N C12CCC(CC1)NC(=O)C(=O)NCCO2.C1(C(=O)OCC)CCCC1CSC CC1CN(C(c2ccc(Cl)nc2I)=O)CCCN1C(=O)CCc1ccoc1 c1(C(=O)NCC(C)N(c2ccnc(C(C)C)n2)C)cc2c(F)ccc(F)c2s1 N1(C(c2nccc(C)c2)=O)C(CNC(=O)Cc2cnc(C)[nH]2)CC2CCCC12 C1(CNC(C#CC(C)(C)O)=O)CCN(C(c2csc(C(F)F)n2)=O)CC1(F)F c1(C(=O)NC(CC=C)C(=O)NCC2(F)CC(CO)C2)cc(C)c(F)cn1 C12CCN(CC1)N2CCOC.n1(CCOC)cc(C(=O)NC2CC2)nn1 c1(C(=O)OCC)ncc(NC(=O)C(=O)NC2CN(C3CCC3)C2)cc1Cl C(=O)(C(C)C(F)(F)C(F)F)N(CCOC)CCNC(=O)C(C)(F)C(C)(C)F CC(O)CCCCCC(=O)NCC1CN(C(=O)C=CCO)CC1C(F)(F)F C1(CNCCC(COC)O)CCCN(C(C)(C)C)C1=O N1(C(c2ccc(CNC(C34CC5CC3C4C5)=O)nc2)=O)CCOCC1CO c1(CC(N2CC(O)CC(NC(CNC(N)=O)=O)C2)=O)ccc(Br)c([N+](=O)[O-])c1 N1(C(c2cc(C)sn2)=O)CCC(NC(C2CCCN(c3nccs3)C2)=O)C(O)C1 C(C(C)(F)C(C)(C)F)NC(C(C)(CO)NC(CC1CC(N(C)C)C1)=O)=O c1(CC(N2CC(OCCNC(CC3CCN(C)C3)=O)C2)=O)sc(O)nc1O c1(C(=O)NCC2CCC(NC(c3nc(C)n(C)c3)=O)C2)nccc2ccncc12 S(=O)(=O)(c1c[nH]ccc1=NC1Cc2cscc2C1)N(CC(C)(C)CO)C CCC(CC)C(=O)NCC(=O)NC(C)C(C)(C)NC(=O)Cc1sccc1Cl c1(NC(CCCC2C(C)C2)=O)cc2cccc(Br)c2cc1O CC1CC(C(=O)NC2CN(C(c3cncc(C(C)(C)C)c3)=O)C2)CCO1 c1(C(N2C(CNC(c3ccnc(O)c3)=O)CC(F)(F)C2)=O)cnn2cccnc12 CC1(CO)CCCC1NC(c1ccc(Cl)s1)=O CC(O)C(C)C(=O)NCC(C1CCCCC1)NC(=O)CC1CN(C)C1 C1(NC(c2c(CC)n[nH]c2)=O)C2CC1CN(C(=O)CNC(c1ccco1)=O)C2 C1(NC(C(C)NC(CC)=O)=O)CCC(O)CN(C(c2cccc([N+](=O)[O-])c2)C)C1 Cc1ccc(C=CC(N2CC(NC(=O)CC3CCCCN3C)C3(CC3)C2)=O)cc1 c1(NC(=O)C(c2ccccc2I)N(CC(F)F)C2CC2)ccc(F)cc1F n1(CC)nc(C(=O)N(CC(C)(C)NC(=O)C(F)(F)C2CCOCC2)C)ccc1=O C=CCCCCCCCCC(=O)N(C1CC2CCC(C1)N2C(=O)CCS(C)=O)C C(=O)(CCCCCNC(=O)CN1CCCCC1)NC(C1CCC(=O)N1)C C[Si](C)(C)C1(CNC(=O)CC2(NC(C34CSCC3C4)=O)CCC2)CC1 c1(OC)cc(C(N2CCC(OCCNC(=O)C(C)(C)OC)C2)=O)cc(Cl)c1OC N1(C(C2(C)COC2)=O)CCC2(CO)CN(C(=O)Cc3ccccc3F)CCC2C1 C=C(C)C1CN(C(C2C3CCC(C3)N2C(c2cccnn2)=O)=O)CCO1 CC(C)CC(C)C(=O)N1CCCCC1CNC(=O)CCSc1ccccc1 C1(NC(C(c2cncnc2)C)=O)CC2CC(C1)N(C(=O)C1=COCC1)C2 N1(C(CC(COC)C)=O)CC(NC(=O)CCCS(C)(=O)=O)CC2(CCOCC2)C1 C1(N(C(c2cnsc2)=O)CC)CCN(C(c2cnc(C(F)F)s2)=O)C1 c1(CNC2CC(C(=O)NC(CC3CCC(C)C3)=O)C2)ncccc1F C1(C2CC2)(CNC(C2CN3CCN2CC3)=O)CCN(C(=O)CCc2cc[nH]n2)C1 N1(C(c2nncn2C)C)CC(NC(c2ncoc2C2CC2)=O)CC2(CCOCC2)C1 n1(C(C)C)cncc1CN(C(=O)C(F)C1CCOC1)C C(=O)(C1CCCn2cncc21)NC1CCN(C(C(=O)NCC2CC2)=O)CC1 N1(C(C(C(C)C)NC(C(COC)(C)C)=O)=O)CC(CO)C2(CC2)C1 C(N=c1[nH]c(-c2ccccc2)nc(=NC)[nH]1)C1N(C(CC=CCC)=O)CCC1 c1(C(N2CCC(CC)C2CNC(=O)C#CC2CC2)=O)c(S(C)(=O)=O)cnn1C C1(C(=O)NC(CC=C)CC)CCC2(CC2)N1C(=O)CC1CC(CC)C1 c1(OCC(N2CCC(NC(C(C(C)C)NC=O)=O)C2)=O)ccc(S(N)(=O)=O)cc1 C1(C(=O)NC2CC(NC(C(C)C)=O)C2)CCCCN1C(C1CCC(C(N)=O)O1)=O N1(C(c2cccc(OCC(F)F)c2)C(=O)NC)CC=CCC12CCOCC2 c1(C(c2n(CCCC)nnn2)NCC2(C)CC2(C)C)cnc(OC)nc1 C12(NC(COCC=CCNC(=O)OC)=O)CCC(CF)(C1)OC2 Cc1ccnc(C(=O)NC(C2CCCC2)CNC(=O)CC2CC2(C)C)c1 C1(C(=O)NCC2N(C(CCS(C)(=O)=O)=O)CC2)CC12C1CC3CC(C1)CC2C3 Nc1cnc(Cl)c(C(=O)NC2CCCN(C(c3cnc(O)c(Cl)c3)=O)C2)c1 c1(CC(C(=O)NCC2(C)CCN(C(CC(=C=C)C)=O)C2)C)ccc([N+](=O)[O-])cc1 CCC(C)C(CC(=O)N1CCCC1COCC)NC(C1CCCC1C)=O Cc1[nH]nc2c1CCC(C(=O)NC1CN(C(C3CN4CCN3CC4)=O)CC1O)C2 C12(Cn3cc(CCN(C(C)=O)CC)nn3)CC1CN(C(=O)Cc1ccc(C)cn1)C2 C1(=CCNC(=O)CC2CC3CCC2O3)CCN(C(=O)CCn2cccc2)CC1 C(=O)(CCCC(C)(C)NC(C1CC1(F)Cl)=O)N(C1(COC)CC1)C Cn1cc(CC(N2CCC(NC(C3CCC3)=O)C2)=O)c2ccccc12 c1(C(=O)NCC2CCCC(NC(CC=C)=O)C2)cccc2c1CCN2 c1(-c2c(OC)ncnc2)ccc(N=c2[nH]cnc3cc(Br)sc23)cc1F C1(CNC(CCSCCC)=O)CN(C(=O)C(=Cc2cccnc2)C)CC(C)(C)O1 C1(N(C(c2coc(CO)c2)=O)CC)CCCN(C(=O)Cc2cccc(C)c2)CC1 c1(OC(C)C(N2CCOCC2C(=O)NC2CCCC2)=O)ccc(C#N)cc1 N1(C(C(CC)OC)=O)CCOCC(C)(CNC(=O)C=CC2CCCC2)C1 C1(N(CC(C)C)C(C2CCCN2C=O)=O)CCN(C(=O)C(C)O)CC1 c1(C(=O)NC2C(N(C)C(c3ccoc3)=O)CCCC2)ccc(F)c2c1CCC2 c1(OC)nccc(-c2cnc(OC)c(C(=O)NCc3ccc(C)nc3)c2)c1F C1(NC(C(C)=C2CC2)=O)COC2(CCN(C(c3cc(C(C)C)ccc3C)=O)C2)C1 C1(NC(=O)NCc2noc(C(C)(C)C)n2)C2CC3C1C3C2(CC)C(=O)O C12(COC)CN(C(C3C(C)OC(C)C3C)=O)C(CO)(C1)C2 C1(NC(CN(C(=O)C(CC(C)C)OC)CC)=O)CC(C)(OC)C1(C)C C1(=O)CCCC(=O)NOCCN1.CCC(C(=O)OC(C)(C)C)C(C)(F)F c1(-c2scc(C(=O)NCCC3(N(C)C)CCC3)n2)ncccc1Cl Nc1cnc(C(N2CCCC2C2(C(c3cccnc3)NCCC(F)F)CC2)=O)cn1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(c2cc(C)c(N)cn2)=O)C2COCC12 CC1CN(C(=O)Cn2cc(CCO)nn2)C(C)C1C.c12ccc(cc1)CNC2=O c1(C(N2C(C)CC(NC(=O)Cc3nc[nH]n3)CC2)=O)csc2c(O)ccnc12 C12CC(C)N(C1)C(=O)C2.C(C(C)(C)C)=CC(=O)N.CC(C)NCCO N1(C(c2c(NC)cnnc2)=O)CC(CNC(=O)C(C)COC(C)C)C2(CCC2)C1 Cc1nc(NCCNC(=O)Nc2cc(-c3c(F)cccc3F)no2)cn(C)c1=O c1(C(=O)NC2C(CC(N3CC(C#CC)C3)=O)C(O)C2)ccn(C)c(=O)c1 N1(C(C2N(C(=O)OC(C)(C)C)CC2)=O)CC2(CCN(C(C3CCCC34CC4)=O)C2)C1 c1(NC(C2N(Cc3c(OC)cccn3)CC(F)(F)C2)=O)ccc([N+](=O)[O-])cc1Br N1(C(c2n(C(C)C)cnc2)=O)CCC(CCN(C(=O)CCC2CC2)C)CC1 C1(CCNC(C2(C#C)CC2)=O)C(C)CCCN1C(=O)CC1(O)CCCCC1 N1(C(=O)C(F)C2CCCC2)CC(C2CCN(C(C3CCC(C)(C)O3)=O)CC2)C1 c1(OCCC(=O)NCC(CC=C)NC(=O)Cc2ccncc2C)ccccc1O C(=O)(CCCCCO)NCc1cccc(CN(C(=O)C(O)CC(F)F)C)c1 c1(C(=O)NC(CNC(c2c(C)csc2)=O)C(C)(C)C)cc2n(n1)CCNC2=O C1(CN(C(=O)C(C)C2CCC2)CC)CCN(C(c2cc(Cl)n[nH]2)=O)CC1 c1(C(=O)NCC2C(NC(C(CC=C)(F)F)=O)C2)cc2c(F)ccc(Br)c2[nH]1 C(=O)(CCCCC(C)(C)OC)N1CC(NC(C(F)=CCC)=O)C(CO)CC1 C12(C(=O)NC(C)CCNC(=O)CC3CCOC3C)CCN(CC1)S(=O)(=O)C2 N1(C(C(COCC)N=[N+]=[N-])=O)CCC(C2CCN(C(C3(C)CC3CC)=O)CC2)C1 N1(C(c2cc(OCC)ncc2)=O)CCC(NC(=O)C2CC2)C(c2ccccc2)C1 c1(N(C(C#C)C)C)nnc(-c2ccc(C)nn2)n1CC1CCCCO1 N1(C(CC(CC2CC2)NC(C(CC)COC)=O)=O)CCOCC2(CC2)C1 C(c1nc(C)cs1)=CC(=O)N(C1CCN(C(C2OCCC2C(C)C)=O)C1)CCC Cc1ccc(C(N2CC(C(C)NC(c3cnc(O)o3)=O)C2)=O)c([N+](=O)[O-])c1 N1(C(C2C(C)CN(C(c3occ4c3CCC4)=O)C2)=O)CCC(CO)C(O)C1 C1(C(=O)OC(C)(C)C)CC(CC(=O)NCCCCc2cnc[nH]2)C1 C1(C(N(C(CCCC)C)C)=O)CC2(CC(NC(C3(CCF)CCC3)=O)C2)C1 C1(C(N2CCC(O)(C(C)C)C2)=O)CC2CCC1N2C(=O)CC(C)(C)C c1(NC)cncc(C(=O)NCC2CN(C(=O)CCc3nc(C)no3)CC2C)c1 c1(C(=O)NC(CNC(COCCC#C)=O)C)ccc(Oc2ccc(F)cc2)cc1 CCCCC(C(=O)N(C(C(=O)NCCNC(=O)C(C)C)C(C)C)C)C(C)C c1(CCC)ccccc1C(=O)NC(C)CNC(=O)COc1ccccc1C N1(C(CCCC(=O)N(C)C)=O)CC2(NC(C3CC(C)(C)CO3)=O)CCC1CC2 c1(C(N(CCC)CCNC(=O)C=CS(C)=O)=O)cccc(O)c1C CC1CNC(=O)CN1C(C1CCCCN1C(C1COCCO1)=O)=O c1(CC)[nH]nc2ccc(C(=O)NCC3CCC(C)N(C(=O)COC)C3)cc12 C(=O)(C(C)CC(F)F)NC(CNC(c1ccc(OCC)nc1)=O)(C)CO C1(CCO)(NC(C(C)O)=O)CN(C(=O)CCCNC(N)=O)C1 C#Cc1cc(C(N2CC3(CC3)CC2CNC(c2sc(C)nc2C)=O)=O)ccc1C C1(C(=O)NC2C3CN(C(c4c(C)ncnc4C)=O)CC32)C2CCC1(C)C2(C)C Cc1cnc(C(=O)NC(C2CN(C(=O)C(F)CC3CCCCC3)CCO2)C)cn1 CC1=C(C(=O)N2CCCC2CCCNC(c2ccc(C)s2)=O)CCO1 CCC(C)(C)CC(=O)NCC1(F)CC(NC(c2cc3scnc3[nH]2)=O)C1 c1(SCC=C(C)C)cc(C(=O)NC2CCCC2NC(=O)CNS(N)(=O)=O)ccc1F O=C(CC1=CCN(C(=O)Cn2c(O)nnc2O)CC1)NC1CCC2(CCC2)C1 C#Cc1cccc(CC(=O)N(CCC(C)NC(=O)CC2CC(=O)C2)C)c1 Cc1n[nH]c(C)c1CC(C)C(=O)NCCCC(C)NC(=O)C=CC(C)(C)C Cc1cc(C)c(C(=O)NC(Cn2cc(C3CCN(C)C3=O)nn2)C(C)(C)C)c(O)n1 c1(C(N2CC(C(C)NC(C(C)SCC)=O)OCC2)=O)ccc2n[nH]c(C)c2c1 C=CCCN=C(NCCn1ncnc1CN1CCC(C)CC1)NCc1ncon1 Cc1nscc1CNC(=O)C(Cc1ccco1)NC(C1CC(=C2CC2)C1)=O c1(CC=CC(=O)NC2CN(C(=O)CCc3cncnc3)C2)ccc(Cl)cc1F c1(C(=O)NC(C)(C)CNC(C2CC2(C)Br)=O)ccc(O)nc1 NS(=O)(=O)c1cc(C(=O)NCC(O)CNC(C2CS(=O)(=O)CC(=O)N2)=O)ccn1 Cc1cc(C)c(C(N2CC(O)CC2CNC(c2nn(C)cc2Cl)=O)=O)cn1 CC(CCCCO)NC(c1cc(-c2ccccc2)n(-c2ccc(F)cc2)n1)=O N1(C(c2cc(C(C)=O)sc2Cl)=O)CCC(c2cccc(C(F)(F)F)c2)C(C)C1 N1(C(CC=C)=O)CC(OC)CC1CNC(c1sc(C)nc1-c1ccc(C)cc1)=O C=C(C)CCCC(=O)N1CCC(NC(=O)C(C)NC(=O)CC(C)(C)C)C(F)C1 c1(C(=O)OC)cccc(CN2CCSCC2C(=O)Nc2cncnc2)n1 c1(C(C(=O)Nc2nc(C(N3CCC(N(C)C)C3)=O)n(C)c2)O)ccc(F)cc1F Cc1ccc(NC(c2occc2CNC(=O)C(C2CCCCC2)C)=O)cc1C C(C(C)(O)CC(=O)NC(CN=[N+]=[N-])C(=O)Nc1ccc(O)cc1OC)OC c1(CC(=O)NCC(CNC(c2c(OCC)ccs2)=O)O)ccc2c(c1)COCC2 C1(C(N(c2cn[nH]c2)C)=O)C2CN(C(=O)CCCn3ccnn3)CC12 CN1CC(N(C)C(C2CN(C(=O)CCc3ccccc3)CCN2C)=O)CCC1=O C(=O)(C(C)(CO)CO)NC1CN(C(c2c(C)cccn2)=O)CC1F N1(C(C2C(C)(C)CCO2)=O)CCC2(CC1)CC(NC(C1(F)CCC1)=O)CO2 C1(NC(C(C)=C2CCCC2)=O)CN(C(=O)CCCc2ccc(O)cc2)CC1C C1(N(C(=O)C=Cc2nccs2)C)CCCC(NC(c2nn(C)cc2Br)=O)C1 C1(C(=O)NCC(=O)OCC2CCC2)CCCCC1N1CCCC1=O C1(C)(CNC(C(F)(F)C2(OC)CCC2)=O)CCCN(C(=O)CN(C)C(C)C)C1 C(=O)(C(O)CCS(C)=O)N1CCCN(C(c2c(CC(=O)OC)ncs2)=O)CC1 c1(NCCC(C)CO)ccc(S(=O)(=O)N2CCC3CCC(C2)S3)c(Br)c1 C(CCO)(C(F)(F)F)N(C(C)C(=O)NC1CCN(C(=O)OC(C)(C)C)CC1)C N1(C(c2cnc(SC)s2)=O)CCOCC(F)(CNC(C2CCCOCC2)=O)C1 N1(S(CCC)(=O)=O)CCCC(NC(CN(CC(=O)OC(C)(C)C)CC2CC2)=O)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCC1(NC(Cc2c(C)n(C)nc2)=O)CC1 c1(C(=O)NC(CC)CNC(C2CCN(CCO)C(=O)C2)=O)cc(F)c(Cl)cc1Cl CCC(CCCC(=O)N1CC(CCO)C1)NC(c1csc(C)n1)=O N1(C(C2C(C)(C)CC2)=O)CCC2(CCCN(CC3CC(C)(C)C3)C2)C1 C1(NC(CSCCCC)=O)(CC)CCCN(C(C2CCCN2C)=O)C1 C1(C(=O)Nc2ccc(O)cc2)(NC(C2CC(OCC)C2)=O)CCCC1C N1(C(c2cc(C)ns2)=O)CC2(CCOCC2)CC1CNC(c1cnc(O)n1C)=O N1(C(Cn2c(C)ccc2C)=O)CCC=C(C(=O)N2CCCC(CCO)C2)C1 c1(OC)ccc(CC(=S)NCCSc2cccc(Br)c2)cc1Br CCCCS(=O)(=O)CC(=O)NCC1CCCC1NC(c1csc(COCCC2CC2)c1)=O C(=O)(C(C)Cc1ccco1)NCCN(C(C1C(CCC)C1)=O)CCOCCOC C=CC(C)(O)CC(=O)NC1CCCC(CC(=O)N(C2CCOC2)CC)C1 C1(C)(C(=O)NCCCNC(C(C)Cc2ccc(F)cc2)=O)COCC1(F)F C1(CC(=O)OC)(OC)CCN(C(C2CCCC2C(=O)OC)=O)CC1 N#CC1(CNC(=O)CN(C(=O)C(O)C(F)(F)F)CCO)CCCCC1 N1(C(C(c2ccc(OC)cc2)CC)=O)CC(N(C(=O)COC)C)C2(CC2)C1 c1(C(C(=O)OCC)N(C)C)ccc(CNC(=O)C(C)CN)cc1.c1(CC)ccn(C)n1 c1(OCC(=O)Oc2ccnn2C(F)(F)F)cc(F)cc(F)c1 C(=O)(C1CCCc2nc[nH]c21)N1CCCCC(CNC(=O)CC2CS(=O)(=O)C2)C1 c1(CNC(C(CC)NC)=O)ccc2c(c1)CN(C(=O)CC1CCCO1)C2 N1(C(c2ccc(C#N)[nH]2)=O)CCC2CC1CN(C(=O)Cc1cc(F)cc(F)c1)C2 C1(CN(C(C)=O)C(C)C)CCN(C(C(=O)Nc2ccc(F)cc2)C2(C)CC2)CC1 c1(C(=O)NC2CC(NC(c3c(C)cn(C)n3)=O)C2)ccc2c(c1)CCC(C)N2 Cc1sc(O)nc1C(=O)NC1(C(=O)NCC2CC(=O)N(C)C2)CC1 C1(NC(c2cn(C=C)nc2)c2nnnn2CC(=C)C)CCCCN(C)C1=O c1(C(=O)NC(C(C)NC(c2n[nH]cc2F)=O)(C)C)cc2c(cn1)OCCC2 CCC(C(=O)NCCCCCCN(C(=O)CCCCOCC)C)C(C)O c1(CC)n[nH]cc1C(=O)NCc1cn(CCNC(=O)CCC2CCC(=O)N2)nn1 N#Cc1cn[nH]c1C(=O)NC1CCC1NC(c1ccc(C(F)F)s1)=O c1(C(C(=O)NC(CC)COC)N(C)C)cccc(Cl)c1 C#CCC(C)(CNC(=O)C(CCF)NC(c1cc(COC)on1)=O)CO c1(CC(C2(C)CCOC2)NC(CC)(C)c2nn[nH]n2)ccc(F)cc1 c1(C2C(C(=O)NCCN(C(=O)CC3(C)CCCO3)CC)C2)ccc(Cl)cc1F c1(C(N2CCCC(CNC(C(C3CC3)OC)=O)CC2)=O)ccc2[nH]ccc2c1 N1(C(C2C(CC)CCO2)=O)CC(C(=O)Nc2cnc(C)nc2C)C(C)(C)C1 CC(C)(C)C(C#N)C(=O)N1CCC(CNC(c2cc3cscc3s2)=O)C1 C1(CCC(=O)NC2CCN(C(c3ccc(C)[nH]3)=O)C2)CCCN(C)C1 C1(NC(CC(C)C(F)F)=O)CN(C(C2CCS(=O)CC2)=O)C2(CCCC2)C1 c1(C(F)(F)F)cc(CSC2CCCC2F)[nH]n1 C1(C(=O)NCc2cc(C(=O)NC(CC#C)C(=O)NC)no2)CC2(CCC2=O)C1 Cc1cnc(C)c(NC(C2CCN(C(=O)CSCC(N)=O)C23CC3)=O)c1 N(C1CSCc2ccccc21)C(C#CC(CNC(C(C)C)=O)(C)C)=O S(=O)(=O)(c1ccc(Cl)nc1)N1CC(F)CC(C(=O)Nc2c(C)ccc(Br)c2)C1 Cc1nnc(CCC(=O)NCCCN(C(=O)C(c2ccccc2)F)C2CC2)s1 C1(C(N2C(C)CCC(NC(c3c(Cl)cc(C)s3)=O)C2)=O)CCc2nncn2C1 CC(CS(C)(=O)=O)C(=O)NC1CC1NC(c1ccc2nccn2c1)=O CCN=C(NCC1=CCCCC1)NC(c1cccc(OC2CCCCC2)c1)OC C(=O)(C1=NOC(C)C1C)NCC(C)CNC(C1Cc2ccccc2C1)=O C12(NC(Cc3cc(C)[nH]n3)=O)CC1CN(C(C1CCS(=O)(=O)C1)=O)C2 Cc1cc(NC(=O)NC(C)CN2CCCC(C)C2)c(F)c(Br)c1 N1(C(CC(C)C)=O)CCC(NC(=O)CCc2cccc([N+](=O)[O-])c2)C2(CCC2)C1 c1(C(N(c2nccc(OC)n2)C2CC3(CNC3)C2)=O)cc2cc(Cl)cc(C)c2[nH]1 C1(CNC(C(CC#C)CC#C)=O)CN(C(=O)C(F)(F)CC)CCC12CCC2 C1(CC(N2CC(O)(CNc3ncc(C(F)F)cn3)C2)=O)CC2CCC1O2 Cc1ncc(C=CC(=O)NC2CCCC(NC(=O)Cc3cn(C4CC4)cn3)C2)s1 C12(CCNC(=O)CC(O)C3CCC3)CCC(C1)N(C(=O)Cc1cncs1)C2 c1(C(=O)NC(C(C)(C)NC(C(C)=C2CC2)=O)C)ccc(N)c(OCCO)c1 C12(C(N3CCC(C)(NC(C(C)n4ccnc4)=O)C3)=O)CCCC(CO1)C2 CC(C)CC(C(=O)N1CCN(C(c2ncccc2O)=O)CC1)n1ccnc1 O=C(CCCCN1CCOCC1)NCCOC1CN(C(C2C3CCCC23)=O)C1 CCC(CC)CC(=O)NCCN(CCOC)C(c1cccc(C2CCCC2)c1)=O Cc1cc(Br)c([N+](=O)[O-])cc1C(=O)Nc1c[nH]nc1C(=O)Nc1[nH]cnc1C#N c1(NCCC2CCC(NC(CNC(CCC)=O)=O)C2)nccc(C(=O)NCC)n1 Cc1cc(C(N2CCC(CC(C)NC(=O)C3=CCCSC3)CC2)=O)cc(C)c1O c1(CC)nc2ccccn2c1C(=O)N(CCCNC(C1C=CC1C(=O)OC)=O)C c1(C(N(C2CC(NC(c3cc(C)ncc3)=O)C2)C)=O)ccc(F)cc1Cl CC1(C)CC(CNC(C2CCOC2CNC(C2(C)CCC(=O)C2)=O)=O)CO1 C(CCC(=O)NC1(C(N)=O)CC=CC1)N(C(C(C)=C(CC)C)=O)C c1(OC)ccc(Br)c(C(=O)NC2CC2NCc2cnc(-c3ccccc3)s2)c1 c1(C(N2CCC(NC(C3CCN(C(C)=O)C3)=O)C23CC3)=O)ccnc2[nH]nnc12 C#Cc1ccc(F)cc1C(N1CC2CC2(NC(c2cnc(SC)nc2O)=O)C1)=O N1(CCNC(=O)CC(F)(F)F)CC2CC1CN2C(c1cc(Cl)ncn1)=O C(=O)(C(C)(C)CCCO)N(CC(C)CNC(c1c(C)nc(CC2CC2)o1)=O)C C1(CNC(C(C(C)C)c2ccncc2)=O)CC2CCC(C1)N2C(C1CC(C)(C)C1)=O c1(NCc2ccc(CC)c(Br)c2)cc(Br)c2c(c1)CNCCO2 c1(CNC(C2CCN(CC(=O)NC)CC2)=O)cc(OC)c(OC)cc1C N1(C(C)C(=O)N(CC(C)(C)NC(=O)Cc2cnn(C(F)F)c2)C)CCCC(O)C1 Cc1[nH]nc2ccc(NC(C3CC3NC(c3ccc(C#N)c(F)c3)=O)=O)cc12 N1(C(C2(C=C)CCC2)=O)CC2CC2(CNC(c2ccc(-n3ccnn3)cc2)=O)C1 c1(C(=O)NC2(C)CN(C(C3(CCOC)CCC3)=O)C2)cccc(Br)c1 C1(CNC(Cc2ccc(CSCC)cc2)=O)CCCN(C(C2CCCO2)=O)CC1 N1(C(CNC(C(CC)C)=O)=O)C(CC(=O)N(CCN=[N+]=[N-])C)C2CCCC12 C1(NC(C(C)NC(C)=O)=O)(CNC(c2ocnc2C)=O)CCOC1 C#CCCC(C(=O)NC(C)C(C)(C)OCC)NC(=O)CN1CCSCC1 N1(C(c2ccsc2Cl)=O)CCC2CCN(C(C3CCn4ccnc4C3)=O)CC2C1 c1(C(N2C(CN(C(=O)C(C)O)CC)CCCC2)=O)ccc(NCC)c2cn[nH]c12 c1(CC(=O)NCCC(C)N(C(=O)C2=CCCC2)C)ccccc1N c1(C(=O)NCCCN(C)C(C2CC23CC(O)C3)=O)ccc2c(c1)SCC(=O)N2 CC1CC1C1CC1NC(=O)C(c1cnn(C)c1)NC(=O)Cc1cccs1 c1(C(N2CCCC(NC(C3CCCC(=O)N3)=O)CC2)=O)ccc2nc(Cl)nn2c1 C1(C(=O)NCCNC(C(CC)CC(F)F)=O)CCc2nc(C3CC3)ncc2C1 C=CCC(C)(C)CC(=O)NC(C1CCN(C(=O)C(C)Cc2cnco2)C1)(C)C C1(C(=O)NC2(CC)CC2)CCN(C(=O)C(c2ccn(C)n2)C)CC1C C12(NC(Cc3ccc(C(C)=O)s3)=O)CCCCC1CN(C(C1(C)CC1(F)F)=O)C2 N1(C(C2(NC(C)C)CC2)=O)CCCCCC(NC(=O)C(=O)NCC2CC2)C1 c1(C(=O)NCC2CC(NC(c3ncn(CC)c3)=O)C2)c[nH]c2ncc(Br)cc12 C#CCC(O)C(=O)NC12CC(C(=O)NC3CCS(=O)(=O)C3)(C1)C2 CC(C)CC(CNC(c1ccc(O)c(F)c1)=O)C(=O)N1CC2CCOC(=O)C12 N1(C(C(=O)NC2CC(=O)NC2)=O)CCC(c2ccccc2)(CO)CC1 C1(C(N(C)CC2N(C(c3n(CC)nnc3)=O)CCOC2)=O)CCCCC12CCC2 C12(NC(=O)NC3CC34CCOCC4)CC(CO)(C1)OC21CCNCC1 C1(C(=O)NCC(C#C)C(C)C)CCCCCCN1C(C1CC2CCC(C1)O2)=O N1(C(C2(c3ccc(C)nc3)CC2)=O)CC(NC(c2n[nH]c(C)c2F)=O)C2(CC2)C1 CCC(CC)(CO)C(=O)NC(CNC(=O)Cc1ccc(Cl)cc1F)SC CC(C)CC(CNC(c1ccc(O)cc1F)=O)C(=O)N1CCCC(CC2CC2)C1 C1(C)(NC(C(Cc2cn[nH]c2)NC(CCSCCCC)=O)=O)CCOC1=O C1(CC(=O)NCCCN(C(c2ccc(CCO)cc2)=O)CC)CCC2(CC2)CO1 c1(C(N2CCC(N(C(c3ccc(C#C)o3)=O)C)C2)=O)n[nH]c2cc(OC)ccc12 CCC(CC)(CCNC(c1cnn(C(C)C)c1)=O)NC(=O)CC1COC(C)(C)C1 CCC(C)(CNC(C1CC2(C1)CC21CC1)=O)C(=O)NC1CCN(C(N)=O)C1 c1(CC)cc(C(=O)N(C2CC(c3ccccc3)C2)C)cc(CC)c1CC(=O)OC N1(C(CSCCC=C)=O)CCCC1.C1C(=O)N1.C1COCCN1C CCCC(C(=O)OC)C(=O)NN=c1cc[nH]cc1OC c1(C(=O)NCCC(=O)NCC(n2ccnn2)C)nc(=N)cc[nH]1 C1(F)(CNC(C(N(C)C)C2CC2)=O)COCCN(C(c2cc(Cl)nnc2O)=O)C1 C1(CNC(c2nc(CC)sc2)=O)CC(COC)CN1C(c1cn(C)cn1)=O c1(COCCOCCOCCNC(=O)CNC(C=C(C)Cl)=O)ccon1 c1(CC(=O)NC2C(NC(C(C(C)C)OC)=O)C2)cc2cccnc2nc1C C1(NC(C2(CC(C)C)CCCC2)=O)CCN(C(C23CC(C)(C2)C3)=O)CC1(C)C CC1=CCN(C(C2CC(N(C(=O)Cc3cc(C)nn3C)C)C2)=O)CC1 c1(OC)cncnc1N1CCCCC1CNC(c1ncccc1Cl)=O C#CCC(C)(C)C(=O)NCC12CC1CN(C(=O)Cc1cccc(C)c1Cl)C2 C1(NC(c2c(CC)nns2)=O)C2CC3C(C2)C13C(=O)N(C)CC1COCCO1 Cc1cnnc(O)c1C(N1CCCC(N(C(=O)C(N2CCN(C)CC2)C)C)C1)=O N1(C(C(C)Cn2cccn2)=O)CCCCC1CN(C)C(C1CC(O)C1)=O c1(C(=O)NCC(CNC(c2c(F)ncc(OC)c2)=O)CO)ccc(C)c(C#N)c1 CC1CCC(OC(=O)Nc2cc(CC(C)(C)C)nn2C(C)(C)C)CC1 c1(C(=O)NC2CCC(N(C(=O)C(=O)NCC3CC3)C)C2)n[nH]c2c1COCC2 N1(C(CC(=O)NCC#C)=O)C2CCC1C(F)C(NC(=O)Cn1ccnn1)C2 C(C1CN(C(=O)C(C)OCCOC2CC2c2ccco2)CC1C(=O)NC)=CC c12cc(ccc1Br)NC2=O.c1(OC)nnc(C2CN(C(=O)CCOC(C)=O)C2)s1 Cc1cc(C(N2CCCC(N(C)C(C3CCS(=O)(=O)CC3)=O)C2)=O)c(O)c(C)c1 N1(C(C2CN(C(CNC(C)=O)=O)C2)=O)CCCCC1C1CCN(C(C)=O)C1 N1(C(CCCCCOC)=O)CCC(NC(c2cnc(C(C)O)s2)=O)C12CCC2 CCCCC(O)CNC(c1c(CNC(C2CC2OC(C)=O)=O)nnn1C)=O C12(C(=O)OC(CCCC)CCC)CCCN1S(=O)(=O)CC2 N1(C(=O)OC)CCOC(c2n[nH]c(C3CC3)n2)C1.C12(C(=O)OC)CC(C1)N2 Cc1ncccc1CC(=O)NCC1C=CCN1C(=O)CCl C1(NC(c2n(C)ncn2)=O)CN(C(=O)Cc2cccc(F)c2F)CC1(F)F N1(C(CCSCCCC)=O)CC2CC(C1)C2NC(c1cccc(OC)c1F)=O C1(C(C)C)(C(=O)NCCCc2cc(O)n[nH]2)CCCN1C(C1CCCCO1)=O Cc1ccnc(O)c1C(=O)NCC(C)NC(c1cn[nH]c1)=O N1(C(CC2(N(C)C)CCC2)=O)CCN(C(C2(C)CC2(F)F)=O)CC12CC2 N1(C(CC2CC(C)C2)=O)CCCC(C)(NC(=O)CCOc2cccnc2)C1 C(C1c2ccsc2CCN1C(C1CC2(CSC2)C1)=O)NC(C1CCN(C)CC1)=O c1(CCC(=O)NC2CC2CNC(C2(C(F)(F)F)CC2)=O)ccccc1F Cc1cc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)Cc2cccc(O)c2)cc1F CC(C)(O)C(F)(F)C(=O)NCc1cc(C(=O)NC2CCC(C)(C)C2)co1 c1(C(N2CC(O)CC(NC(C(CCC)CC)=O)C2)=O)cc2c(=O)[nH]ccn2n1 CC1CN(C(=O)C(F)OC(F)(F)F)CC1n1cc(CC2(O)COC2)nn1 N1(C(c2c(C)n[nH]c2C)=O)CCC2(CC1)CC(CNC(=O)C1=CCCC1C)C2 c1(C(=O)NC(C2(CNC(C(CC)C)=O)CC2)C)nc(C(C)C)ncc1Br CCC(CC(=O)N(CC(=O)NOCc1ccccc1)C1CCCC1)OC COn1cnc(C)c1C(=O)NCC(C)(C)OCCNC(c1cncn1C)=O C1(C(=O)NC(C)CNC(=O)CC23CC(C2)C3)CCOC2(CCCC2)C1 C1(NC(CCC2(N)CCC2)=O)CC(CO)C2CC12.C(CC(CC)C)=CC c1(OC)ccccc1CC(=O)NC(C)C(C(C)C)NC(=O)CN(S(C)(=O)=O)C C=CCC(CC(=O)N1CCCC1CCOC)NC(C1CN(C(N)=O)C1)=O c1(Nc2cc(Cl)c(I)cc2)cnc2c(Cl)ccnn12 c1(N2CCC(NC(C)=O)C2)[nH]c(=NCCN2CCCCCC2)nc2ncn(C)c12 C(C)(CCC(=O)NCC1CCCCN1C(c1cc(C2CC2)ncn1)=O)OC N1(C(C=CC(=O)N(C)C)=O)CCCC2(CNC(=O)Cc3cscn3)CCCCC12 C1(CNC(CC(C(C)C)C)=O)CCC2CN(C(c3cc(Cl)cn3C)=O)CC12 N1(C(C(CC)SC)=O)CC2CCCCC2(CNC(=O)CCCn2cncn2)C1 N1(CC(=O)NCC(C2CC2)NC(C2(C(F)F)CCCO2)=O)CC2CC2C1 N1(C(Cn2c(C)ncc2)=O)CCC2(CCO2)C1.C12CCC(CC1)C(=O)N2 Cc1c(CC(=O)NCCN(C)C(C2(C(F)(F)F)CC=CC2)=O)cnn1C C1(C(=O)NCc2c(C#C)cncc2)CC12CCN(C(c1cccc(Cl)n1)=O)CC2 c1(C(N2C(C)CC(NC(=O)CCC(C)CN(C)C)C2)=O)c(O)nnc2c1CCC2 C1(C2CCCN(C(=O)C(F)C3CCC3)C2)(NC(=O)CC2CCC=CCC2)CC1 N1(C(C2N(CC)CCCC2)=O)CC=C(CNC(c2c[nH]nc2C(C)C)=O)CC1 CCC(C)C(C(=O)OC)NCC12CC(CC(C)O1)C2.C1(=O)CN1 c1(C(=O)NC(C(N2CC(CC)(OC)C2)=O)Cc2cc[nH]n2)ccc(C2CC2)cc1 C#CC1CN2N3CCC(OCCCO)(C3)OC1C2.C(C)(C)(C)OC(=O)NC Cc1nc(N)cnc1C(=O)NC1(C)CCCN(C(=O)CSc2cccc(F)c2)C1 CC(O)CC(CN(C1CCCC1)C(=O)NCCC#N)c1ccccc1 N1(C(C2N(CC)CCOC2)=O)CCCC2(CCN(C(c3csnc3Cl)=O)C2)C1 C1(C(=O)NCC(CC)(C)CC)CCN(C(=O)CCN(C)C)O1 N1(C(c2c(C)cc(CC)o2)=O)CCOC2(CCCN(C(C3(C)CCCC3)=O)C2)C1 c1(CC(=O)N(C(C)C)C2CC2)ccc2c(c1)CN(C(c1cnc(O)[nH]1)=O)CC2 N1(C(C)=O)CCOC(C(N2CCCC2C2(NC(C3CC(Cl)(Cl)C3)=O)CC2)=O)C1 C(=O)(C1=C(Cl)CCOC1)N1C(C(C)(C)NC(=O)CS(F)(F)(F)(F)F)CCC1 c1(C(=O)NCC2C(NC(CC(C)c3ccncc3)=O)C2)[nH]nc2c1CCC2(C)C C1(CNC(C=CC(C)NC(C2(SC)CC2)=O)=O)(CO)CC2CC2C1 c1(C(N2C(CNC(=O)C3=CCCCO3)CC(OC)C2)=O)cc(C)c(Cl)cc1F N1(C(COC)=O)CCCC(C)C1CNC(=O)Cc1ccc(Br)cc1Br C(=O)(CC(C)(C)CC(=O)NCC(c1ccccc1)NC(c1csnc1C)=O)OC N1(C(C=CCCC)=O)CC(C(=O)NCC(O)CCOC)CC(C)(C)C1 Cc1cc(F)c(N)cc1C(=O)NC(C)CCCNC(c1occ2c1CCOC2)=O N1(C(CCC(CC)C)=O)C2CCC1CC(C(=O)NC1CCN3CCC1C3)C2 N1(C(c2c(C)noc2C)=O)CC2(CCC(C(=O)NC(C)C#N)O2)C1 C12CCC(CC1)C(=O)NC2.C1(NC(C=CCC)=O)CC(CC)(CC)C1 C1(O)(CCNC(CCC=CC(C)C)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1 C1(NC(C2CCCN(C(C)C)C2)=O)CC12CCOCC2 c1(C(=O)NCCCN(C)C(C2(CF)CCC2)=O)nn(C(C)(C)C)cc1[N+](=O)[O-] c1(CC)conc1C(=O)N(CC(CC)NC(=O)CN(C)C(N)=O)C C1(C(=O)NC2C3CN(C(C4C(C(N)=O)C4)=O)CC2C3)CCCC2(C1)CC2(F)F c1(C(N(CCOC)CCNC(c2cnc(O)s2)=O)=O)cn(C)c(=O)cc1C c1(C(=O)N(CCCN(C2CCCC2)C)C(C2(C)CCCO2)=O)ccc(C(F)F)cn1 c1(CC(N2CCC(C(CN(C(C(C)C#N)=O)C3CC3)O)CC2)=O)cccc(F)c1F N1(C(c2ccc(C(C)=O)s2)=O)CC(N(C)C(c2cn(C)cn2)=O)C(C)(C)C1 N1(S(c2n(C)ccn2)(=O)=O)CCc2sccc2C1c1ccccc1 N1(C(c2cccnc2F)=O)CC2CCC(C1)C2NCc1ccc(Cl)c(F)c1 C1(C(=O)NCC2C(NC(C(c3ccnn3C)C)=O)CC2)CCCN1C c1(OC)ccnc(C(=O)NCCCCn2cc(C(C)(C)C)cn2)c1C CS(=O)(=O)c1coc(CN2CCC(CCNC(=O)CCCc3ccccc3)C2)c1 CCC(CC)CC(F)C(=O)NCCOCC(N1CCC1CN(C)C)=O C(=O)(CC(C(F)(F)F)NC(C1CC2C=CC1C2)=O)NC(CCC)c1ccco1 C1(CC(=O)NCC(CO)NC(C(C)=C2CC2)=O)CCN(C)C1=O C#Cc1cc(C(N2CCC(N(CCC)C(c3scnc3C)=O)CC2)=O)cc(F)c1 c1(C(n2cc(C3CCCN3C(=O)Cn3cccn3)nn2)C)cccc(N(C)C)c1 C(=O)(C(C(C)C)C(C)C)NC(c1cnn(C)c1)C(=O)NC(c1c(C)ncs1)C CCCC(C)C(=O)N1CCCCC1C(=O)NCc1nocc1C(C)C C1(NC(=O)CCNc2ccccc2)CC2(C1)CC2NC(=O)COC1CCCC1 C(=O)(C1=CCc2ccccc21)N1CC2C(CNC(C(CCCC)F)=O)(C2)C1 O=C(CCN1C(=O)COc2ccccc21)NC1CCOC2(CCSCC2)C1 c1(OC)cc(C(N2CC3CN(Cc4cccc(Cl)c4)C3C2)=O)cc(O)c1O C(=O)(CCCS(N)(=O)=O)N1C(C2(C(C)(C)CNC(=O)C=CC3CCC3)CC2)CCC1 C1(CCOC)(NC(C2CC2C(=O)OC)=O)CCN(C(C2CC=CCC2)=O)C1 c1(CNC2CC(NC(C3(C)CCCC3)=O)C2)ccc(Br)nc1Br c1(C(N2CC3CN(Cc4nc(C)oc4)CC3C2)=O)cccc2cccnc12 c1(CC(=O)NCC2(C)N(C(c3c(COC)cco3)=O)CCC2)ccc(O)c(F)c1 c1(C(=O)NC(c2cccnc2)C(=O)NC(CC(C)O)C)cnc(O)c(F)c1 C(CN=c1cc(C)c(S(=O)(=O)N2CC(O)C(C)(C)C2)c[nH]1)c1cc(C)on1 N1(C(C2C(C)(C)OCC2)=O)CCC(C(F)(F)F)C(NC(=O)CCC2CCC2)C1 c1(OC)ccc(Br)c(F)c1CN1CCC1C(=O)Nc1ccc(O)nc1 C#CC1(NC(C23COC(C2)C(NC(=O)CCc2cc(C)on2)C3)=O)CC(F)(F)C1 C(=O)(CC(O)CC(C)(C)C)NCCC(CNC(C1CC2OC1C1CC21)=O)OC N1(CC(N2C(CCNC(Cn3c(C)cnc3)=O)CCC2)=O)CCC(O)CC1 CC1(C(=O)NC2CCCN(C(=O)CCc3cccc(O)n3)C2)CCCCO1 C1(CNC(=O)C(=O)N2CC(Cc3cccnc3)C2)CCCCC1O C1(C)(CNC(Cc2cncc(C)c2)=O)CCCN(C(c2ccc(N)c(O)n2)=O)C1 N1(C(Cc2ccc(C)s2)=O)C2CCCC1CN(C(c1ccns1)=O)CC2 c1(CC)nn(C)c(C(=O)NC2CCC(CCNC(=O)CC3OCCO3)C2)c1Cl S(=O)(=O)(c1cnc(NCCCC2CCOC2)c(Cl)c1)N(CCCCO)C CCC(C)(C)C(O)C(=O)N1CCC(CNC(c2ccc(SC(F)(F)F)s2)=O)CC1 c1(NC(=O)OC)ccc(F)cc1C1(O)CN(C(=O)N(C(C)(C)C)C)C1 c1(NC)cccc(CCC(=O)NCC(F)CNC(=O)C(C)(C)n2cnnn2)c1 C(=O)(C(C)(C)CS(N)(=O)=O)NCCOCCCNC(C(C(C)C)C#N)=O C1(F)(C(=O)NCCOCCCN(C(C(C)N(C)C)=O)C)CC12CCCCC2 C1(COC)(CNC(C2CC2(C)C)=O)CCN(C(=O)CN2CC3CC3C2)CC1 C1(C(=O)NOCC2CCCCC2)(CC=C)CCCN1C(c1cnncc1C)=O CC(C)CCCCCCC(=O)NC1CN(C(=O)C(C)NS(C)(=O)=O)C(C)(C)C1 N1(C(C2(OCC)CCCC2)=O)CC2(CCC2NC(=O)C=CCF)C1 c1(N2CCC(C3(C)CC3)C2)nc(=NCC23CC(CCO2)C3)[nH]c2cc[nH]c12 C1(C(C)(C)C)CN(C(=O)CNS(N)(=O)=O)CCN1C(=O)Cc1cc[nH]n1 C1(NC(C(N(C)C)C2CC2)=O)CCCC1NC(=O)CC1(C#N)CC1 CC(CC(=O)NCCC1CCN(C(=O)CNC(C2CCCC2)=O)C1)P(C)(C)=O c1(CNC(c2c(CNC(C3C(C(=O)OC)C3)=O)noc2)=O)ccc2ncoc2c1 C1(C(=O)NCC2CC(NC(=O)CC(C)N3CCCC3=O)C2)(OC)CCOCC1 C(c1c(C)noc1C)=CC(=O)NCC1N(C(c2c(C)cc(C)o2)=O)CCC1 N1(C(C2C(c3n(C)ccn3)C2C)=O)CC(O)(C2CCN(C(=O)C(O)C(F)F)CC2)C1 c1(CC)sc(=N)[nH]c1C(=O)NCC(C)CN(C(=O)CCc1nccs1)C N1(CC=C)CCCC(NC(c2ccccc2)=O)C1C c1(C(N2CC(CC)N(C(=O)C=CCO)CC2)=O)cnc2c(c1)CCOC2 c1(C(N(C2CN(C(C(C)SC)=O)CC2F)C)=O)ccc2c(c1)NC(=O)CO2 C(=O)(C(C)CCC(C)(C)C)NC1(CNC(C(COCC)C)=O)CCOCC1 CC#CCC(C(=O)NC1C=NNC1=O)n1cc(Cc2sc(C)cc2C)nn1 c1(C(=O)NC2CC(NC(C(CCOC)OC)=O)C2)cc2nc(=O)ccn2[nH]1 N1(C(C2C3CN(C(C4C(C)CCO4)=O)CC32)=O)CCOC(C)(C)C1 C1(CNC(C(CCSC)O)=O)CCC2(CN(C(=O)CNc3ccccn3)C2)O1 c1(C(=O)NC(C2CC(NC(=O)C(c3cccnc3)O)C2)C)ncn2ccccc12 N1(C(C2C(C)(C)CN(C(C3C=CCS3)=O)C2)=O)Cc2cncnc2C1 c1(-c2nc(CC(CC)C)nn2CCc2ccccc2OC)cnn2c1CCCC2 C1(C)(CNC(CNC(CC)=O)=O)CC(NC(=O)C=CC(C)(C)SC)C1 c1(OC)nc(Br)cnc1NC(=O)CC1CCC(NC(=O)Cn2ccnn2)C1 CC(C)C(Cc1ccccc1)C(=O)Nc1ccnn1-c1cccnc1 C12(C(=O)NCCC3N(C(c4scnc4C4CC4)=O)CCSC3)CCCC1C2(F)F c1(C(C)C)cc(=NCCCCC(C)NC(C2CC3(CC3)C2)=O)[nH]cn1 C(=O)(CN=S(C)(C)=O)NCCC1(C)CCN(C(c2cnn(C(CC)C)c2C)=O)C1 c1(CCNC(=O)NC2CC(C(=O)OC)CN2C)ccc(OC)cc1OC c1(CC)[nH]c(C(=O)NC(C)CN(C)C(c2cc(C(F)(F)F)cs2)=O)nc1Cl C1(NC(c2cccc(C(=O)NC3CC3)n2)=O)CC2CC1N(C(C1CC1(Cl)Cl)=O)C2 N1(C(c2c(CC)noc2)=O)CCC2CN(C(=O)CC3SC(=N)NC3=O)CC2C1 c1(Cc2nnc(C(C(=O)N(CC(C)(C)CN(C)C)C)N(C)C)s2)ccc(Cl)cc1 c1(CNCCCOc2c(C)cccc2Br)ccc2[nH]ccc2n1 CC1(CNC(=O)CNS(N)(=O)=O)CCCN(C(=O)C(c2ccccc2)C2CC2)C1 CCC(F)(F)CC(=O)NCC1(CNC(C2(C)CSC2)=O)CC12CCC2 CCC(C(=O)NCC1CCN1C(=O)C(n1cc(C)cn1)C)NC(N)=O Cc1[nH]nc2ncc(C(N3CC(CNC(c4cc(Cl)cs4)=O)C4CC34)=O)cc12 CN1CCN(C(=O)CCn2ccnc2)CC1CNC(=O)C(O)P(C)(C)=O c1(C(C2COC2)C)n[nH]c(C2CC2)n1 C1(C(C)NC(c2cc(C)ns2)=O)CN(C(=O)Cc2cnccc2C)CCO1 c1(C(=O)NCCNC(C=Cc2cncc(OC)c2)=O)c(Cl)cc(Br)cc1Cl C1(N(C(C2CC(OC)C2)=O)C)CN(C(=O)CCS(N)(=O)=O)CCC1C Cc1ccc(C(=O)NCC2CCN2C(c2ccc(Cl)c(Cl)c2)=O)c(N)c1Cl C1(C(=O)NC(C)CNC(C2CC2C)=O)CCC(=O)N1Cc1ccccc1 CCC1=NOC(C(=O)NC2(C(=O)NC(c3ncn(C)n3)C)CCCC2)C1 C1(C)(NC(C)=O)CCN(C(=O)CN(C(=O)CC2C(C)(C)C2(C)C)C2CC2)C1 CC1CC(CNC(=O)CCCC2CC2)CCN1C(C1CCC2(CCC2)C1)=O C1(C)(C(=O)Sc2cccc(C)c2)CCCN(C2CCCC2)C1.C1(=O)C(C2CC2)N1 Cc1cc(C(=O)NC(CNC(c2cnc(O)s2)=O)C(C)C)no1 c1(N2C3CCC(CN(C)C)(CC3)C2)nc(=NCCC2=NOCC2)[nH]c2c1SCC2 S(=O)(=O)(c1cnc2c(Br)csc2c1)NCCS(N)(=O)=O N1(C(c2c(OC)cc(F)c(F)c2)C(=O)NC2CCC2)CC2CS(=O)(=O)CC2(C)C1 c1(C(=O)N(CC2CC2)CC2CC2)cc2sccc2[nH]1.C12CCN(CC1)C2 C(C(C)(CC(=O)NCC(C1CCC1)NC(=O)C(C)(C)O)C(F)(F)F)N(C)C n1(CCSC)nnnc1C(C)(CC1CCCO1)NC(C)C C(CC(=O)NCC=CCNC(C1CC2(C1)CC(O)C2)=O)(C(N)=O)NC(C)=O c1(CCOCC(=O)NC2(CN(C(=O)CC3CCCCO3)C)CC2)ccc(Cl)s1 C1(CNC(C2N(C(C)=O)CCC2)=O)CCCC2CN(C(C3CC3COC)=O)CC12 c1(-c2nnc(N3CC(OC)CC(CC)C3)n2CCOC)cc(F)c(F)cc1Cl C12(NC(c3cncs3)=O)CCCC1N(C(c1nnc3ccccn13)=O)CC2 c1(C(=O)NC(CC)CNC(C2CCCC(O)C2)=O)nc(C(C)C)ncc1Cl Cc1ccccc1COCC(=O)NC(C)CN(C)C(c1coc(C2CC2)c1)=O c1(C(=O)NC2CCC2CNC(c2c[nH]nc2[N+](=O)[O-])=O)cc2ncccn2n1 c1(OC)cc(OC)c(C(=O)N(CC(O)CNC(=O)C(C)NC(C)=O)C)c(N)c1Cl C(C(C)(C)CCNC(=O)COCCCF)NC(Cn1ncc(C)c1)=O c1(CNC(=O)NOCC2CC2(Cl)Cl)cccc(Cl)c1 N1(CCCC(=O)NC(CNC(C2C(C=C)C2)=O)(C)C)C(=O)c2ccccc2C1=O C1(CNC(C(C=C)(F)F)=O)CC12CCN(C(=O)CSc1nnnn1C)CC2 c1(Cc2nc(C(=O)Nc3cc(OC)ncc3C)sc2)ncnc2[nH]cc(C)c12 N1(C(C)=O)CCCCC1C(=O)NC1CN(C(=O)C(N)=O)C1 C1(NC(c2c(C)nn(C)c2)=O)CN(c2cc(C(N)=O)nc(Cl)n2)C2CCCCC12 c1(C(=O)NC(CC=C)CNC(c2cc(C3CCOCC3)on2)=O)cncc(C)n1 CS(=N)(=O)C1CN(C(C2(NC(C3CC4(CCC4O)C3)=O)CCSC2)=O)C1 c1(N2CCC(CC(=O)NC3CCCCO3)C2)ccc(CO)cc1F N1(Cc2ccc(CC(=O)O)cc2)CC2(CCN2C(=O)CCc2ccccc2Cl)C1 c1(OC)ccccc1SC(C(=O)N(C1CN(C(c2ccc(SC)cc2)=O)C1)C)C c1(C(CC(=O)NCCCCCCNC(CC(=O)OCC)=O)O)ccc(Cl)c(Cl)c1 N1(C(CCCN(C)C)=O)CCCC(N(C(=O)CSC(C)(C)C)C)C1 C(=O)(C(C)(O)C(F)(F)F)N1CC(CNC(CC(C=C)(C)C)=O)OCC1 C1(C)(CC(=O)NC(C2CCCC2)CNC(C(C)CF)=O)CCS(=O)(=O)N1 C1(C2(NC(c3ccsc3)=O)CC2)CCCCN1C(c1cc(C(F)(F)F)ccn1)=O c1(CNC(CCOCC#C)=O)ccc2c(c1)CN(C(c1sc(CO)nc1C)=O)C2 CCCCCC(O)C(=O)NCC1CCN(C(c2sccc2Br)=O)C1 C1(C(N2C(CN(C(=O)Cc3cnc(C4CC4)[nH]3)C)CCC2)=O)CCCCNC1=O c1(C(=O)NC2(CCCNC(C(=O)NCCOC)=O)CC2)cn(C)c(=O)cc1C c1(CNC(c2c(COC)ocn2)=O)cccnc1F c1(NC(c2ncc(C)[nH]2)C2CCC2)ccc2c(c1)nnn2C C1(NC(Cc2ccc(OC)c(F)c2)=O)CN(C(C2CCOC2)=O)C2(CCCC2)C1 C(C(=O)N(C1CN(C(C2CC2C(F)(F)F)=O)C1)CCO)(C(C)C)OCC C(CO)(C(O)C1CCC1)NC(=O)C(=O)N1CCC1C1CCC1 c1(C(N2CC(N(C)C(C34CCC(F)(CC3)C4)=O)C2)=O)cc2c(nc1O)CCSC2 C1(NC(c2c(C)c[nH]n2)=O)CC(O)CN(C(c2cc(Cl)cnc2O)=O)C1 N1(C(COC(C)C)=O)CCC(C)(NC(=O)CCCc2ccccn2)CC1 N1(C(c2ccc(C)o2)=O)CC2(CCN(C(C3CC3Br)=O)C2)C1 Cn1cnn(CC(N2CC(O)(CNC(c3ccc(F)nc3)=O)C2)=O)c1=O C1(NC(C(C)NC(CC)=O)=O)CCCCC1NC(C1CC(=O)N(C)C1)=O C1(NC(CCS(N)(=O)=O)=O)CN(C(c2ccc3ocnc3n2)=O)CC12CCC2 c1(C(=O)NCC2N(C(=O)CC3=CCCC3)CCN(C)C2)n[nH]c2c1CCSC2 Cc1ncnc(C)c1C(=O)NCC1(C)CCCN1C(C1C=CC=CC=C1)=O C1(C(N(CC(C)NC(c2nonc2N)=O)CC)=O)CCOC(CC)C1 c1(C(N(CC(C)N(C(C(C)C2CCOC2)=O)C)C)=O)ccc(C(F)(F)F)c(F)c1 C(c1ccc(O)cc1Cl)=CC(N1CCC(C)(NC(COCCOC)=O)C1)=O N1(C(C(COC)N(C)C)=O)CCC(CNC(=O)CCCCl)C12CCC2 C=C(F)C1(CC(=O)NC2CC2C(=O)N(CC(C2CCC2)OC)C)CCC1 C(=O)(CC(C)C(F)(F)F)N1CC(C)OC(C(=O)N(C)Cc2cocn2)C1 c1(CC(=O)NC23C(NC(C=COCC)=O)CC(CC2)C3)ccc(Cl)c(C)c1F C1(C(=O)NCC2(F)CC(CNC(C3C(N(C)C)CCC3)=O)C2)CCCC(O)C1 C(=O)(C(CC1CC1)NC(C1(CF)CC(=O)C1)=O)NCC(C)CC1CC1 c1(CCC)ccc(C(=O)NCC2CCN2C(=O)CN2CC=CC2)cc1S(N)(=O)=O c1(C(=O)NCC(O)CNC(C2CC3CC3C2)=O)csc(Cc2ccccc2)n1 Cc1ccc(C(F)(F)C(N2CC(O)CC2CNC(c2ccco2)=O)=O)cc1 c1(N2CCCC(NC(C(COC)(C)C)=O)C2C)nc2ccc(Br)cc2s1 Cc1cnc(C(N2CCC(CN(C)C(C3CC4CC4C3)=O)C2)=O)cc1C c1(C(C)C)ccccc1CC(=O)NC1CC1CNC(c1c(Br)nnn1C)=O C1(NC(C=CC)=O)CN(C(c2ccc(F)c(C)c2O)=O)CCC12CCC2 c1(C(N2CC(NC(C3C(F)(F)C34CC4)=O)C2)=O)ccc2c(c1)S(=O)(=O)NC=N2 c1(OC)ccccc1C(C)(C)NC(=O)NC1CCOC(c2ccnn2C)C1 C(=O)(CC(C)C(F)(F)F)N(C(C)CCNC(c1ccnc(Cl)c1N)=O)C C1(NC(C(F)=CCC)=O)CC(O)CN(C(c2scc(C)c2OC)=O)C1 N1(C(C(N2CCCC(C)C2)=O)=O)CCC2(CCOCC2)C(NC(c2nccs2)=O)C1 N1(C(COC)=O)CCN(C(C2CCCOC2C)=O)C(C)C1 C=CC(C)(CC)C(=O)NCc1cc(O)nc(CNC(=O)C(CCC)OCC)n1 Cc1ccc2c(c1)CCC(C(=O)NCCCC(C)NC(=O)Cc1ncc(C)s1)O2 c1(OCC)cccc(F)c1CN1CCCC1C(=O)Nc1cccnc1C N#Cc1ccc2c(c1)CCCC2C(=O)NCCCCC(CO)NC(=O)C=CCF C(N=c1cc(C(C)C)nc(CC)[nH]1)C1C(NC(CNC(C(CC=C)C)=O)=O)CCC1 c1(C(N2CCC(OC)(CNC(=O)C(C)O)CC2)=O)cc(F)c(Br)c(F)c1 C1(NC(c2coc(C(F)F)c2)=O)CC(CNC(=O)C(C2CC2)C2CC2)CC1O C12(C(=O)NCC(CNC(Cc3c(C)noc3Cl)=O)(C)C)OCCCC1C2(F)F C1(C(=O)OC)CCN(C(=O)C2(F)CCN(C(=O)Cc3ccsc3)C2)O1 c1(C(C(=O)N(C(CNC(C(=O)OC)=O)C)C)(F)F)cccc(C(F)(F)F)n1 Cc1cc(=N)[nH]c(C)c1CNC(N1CC(CNC)C2(CCC2)C1)=O N1(C(C2(C)ON=C(C)C2)=O)CC2CC(NC(=O)CCN(C)CCO)CC2C1 c1(OC)ccnc(C(=O)NC2CC(F)(CNC(C3(C(C)C)CCC3)=O)C2)c1F CC1CC(=O)NC1C(N1CC(OCC(=O)NC2COCCC2O)C1)=O N1(C(=O)CCCn2cccn2)CC2(C1)CN(C(=O)CS(=O)(=O)C1CC1)CC2CO c1(C(=O)NC2CCCC(NC(c3ccc(NC)cc3)=O)C2)c(C)ncnc1O CC1(C)CC(NC(c2nc(C3CC3)cs2)=O)CCN(C(=O)CCC2CC2(C)C)C1 c1(OC)cc(C(N2CCCC2)=O)on1.C(=O)(CNC1CC1)NCCC1(C(=O)OC)CC1 S(=O)(=O)(c1ccc(C#N)c(NC2CCC2N(C)C)c1)NC(C)Cc1nncn1C C1(C(=O)NCC2(COC)CN(C(=O)CC(C)N(C)C)C2)CCC2(CCC2)CO1 C=CC(C)(C)C(=O)NCC1C2CN(C(=O)CCc3cccnc3)CC12 c1(-c2cn(CCc3nc(C(=O)OC)sc3)nn2)c(F)cc(OC)cc1Cl C1(CNC(CCN2CCN(CC)CC2)=O)CC2CCC1N(C(=O)C(F)F)C2 N1(C(c2c(OC)nccc2C)=O)CCCC2CN(C(=O)Cn3cncn3)CC12 Cc1cc(-n2nc(-c3cscn3)nc2-c2cscc2C)cc(C)c1 C#Cc1cn(C)nc1C(N1CC(CCC(=O)NOCC(=O)N(C)C)(C)C1)=O N1(C(c2c(C)scn2)=O)CC2(C1)CN(C(c1c(C)noc1C(C)C)=O)CCO2 N1(C(c2n(CC#C)cnn2)=O)CCC(CNC(C23CC4CC2C3C4)=O)CC1 c1(CCC(N2CC(F)(CNC(C(C)OCC(C)C)=O)C2)=O)cccc(O)c1 C1(C(N)=O)(CNC(C2C(C(N)=O)CC2)=O)CN(C(C2CCC(=O)N2)=O)C1 c1(C(N2CC3C(NC(C4CN(CCC)C(=O)C4)=O)C3C2)=O)cc(C)c(C)c(F)c1 N1(C(C2CC(C)CC(C)C2)=O)CCC(C)(C)C(NC(=O)C(N2CCSCC2)C)C1 C1(NC(c2c(C)n[nH]c2C)=O)CN(C(C2(C)CCSCC2)=O)CCC12CCC2 c1(NCC)cnc(C(c2nnnn2CCCF)Nc2cc(C(C)C)nn2C)cn1 C(C(CC1CCCC1)C(=O)NCC1CC1Cl)NC(=O)Cc1cn[nH]c1 CC(C(=O)N1CCOC(CCCNC(C2(c3nccs3)CC2)=O)C1)S(N)(=O)=O N1(C(c2ccc(C#N)c(Cl)c2)=O)CCC2(CCC2)C(NC(C2CC=CCO2)=O)C1 N1(C(CN(S(C)(=O)=O)C)=O)CC2(C(=O)NCc3cccnc3F)CCC1CC2 Cc1cc2cc(NC(C3CN(c4nc(Cl)nc(C)c4Cl)CCO3)=O)oc2cc1C c1(C(C(=O)NC(CC=C)CNC(=O)CC2(C)CCC2)C)ccccc1C(F)(F)F C(c1c(F)cccc1F)=CC(=O)NCC(C(C)C)NC(c1coc2c1CSC2)=O c1(C(N(CC(CNC(C2(C)CCN(C)C2=O)=O)O)C)=O)cnc2sccn2c1=O c1(CC(=O)NCC(CC=C)NC(C23CCCC(C2)OC3)=O)ccc2c(n1)OCCO2 C1(NC(c2c(OC)n[nH]c2)=O)C(C)CN(C(c2[nH]c(O)nc2C)=O)CC1C c1(C(=O)OCCCCC2(C)ON=C(C)C2)cc(C)c(C#N)c(C)n1 Cc1cc(C(=O)NC2COCC2n2cc(C(C)(C)C3CC3)nn2)ncc1Br C=C1COCCN(C(=O)CN(C(=O)C(C)Cn2cccn2)C2CCC2)C1 C1(C(=O)NCC(C)(C)OCCNC(C=CC(C)C)=O)CC2C=CC1C21CC1 c1(C(N2CCC(CC(N3C(CC)CN(C)CC3)=O)C2)=O)ncc2c(ncn2C)n1 CC(C)CCCCCC(=O)N1CCOC(CCCNC(C2CC2C(C)(F)F)=O)C1 C1(C(=O)NCC2ON=C(C)C2)CCN(C(=O)C2(Cl)CC2)O1 C(=O)(C(CSC)NC(C1COCC1N(C)C)=O)NCC(CC1CC1)OC N1(C(C2C(C)(C)C2)=O)CCCC1C1(C(=O)Nc2cc(C(N)=O)[nH]n2)CC1 C1(CC#C)(C(=O)N(CC(O)CN(C(=O)Cc2cncn2C)C)C)CCCCC1 C12(NC(c3c(OCC#C)nccc3)=O)CCC1CN(C(c1cc(CC)c[nH]1)=O)C2 C1(NC(c2coc(Cl)c2)=O)(CO)CCCN(C(C2(c3ccccc3)CC2)=O)C1 N1(C2CN(C(CC3CC(=C)C3)=O)C2)CCN(C(=O)Cn2nccc2C)CC1 CCC(CC)CC(C(=O)NCc1ccco1)N1CCOC(CC)C1 N1(C(C=C(C)C(F)F)=O)CCCCC(NC(=O)CC2OCCCC2(C)C)C1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC2C1CCCN2C(C1CCC(CO)CC1)=O c1(NC(CCNC(C2(C=C)CCC2)=O)=O)cnc2[nH]ncc2c1 N1(C(CCC(C)(C)F)=O)CCC2CN(C(c3cc(C(N)=O)[nH]n3)=O)CCC12 C1(F)(CNC(CCC(C)OCC)=O)CCC(CNC(=O)Cc2cnn(C)c2)CC1 c1(C(=O)OC)nc(=NC2COC3(CCN(C(C4CCOC4)=O)CC3)C2)c(F)c(Cl)[nH]1 CC(C)(C)CCCCCC(=O)N1CCC(CNC(c2c(O)cccc2F)=O)C1 C1(C)(CC(=O)N(CCCNC(=O)C(O)C(F)F)C(C)C)CCS(=O)(=O)N1 CN1CCCC(CC(N2CCOCC2CNC(C2(C)CCSCC2)=O)=O)C1 C=C=CCCC(=O)N(CCNC(C1CCCC1C)=O)CC Cc1ccc(=N)[nH]c1C(=O)NC1(CNC(C2CCCN2C2CCCCC2)=O)CC1 N1(CCC)CC(C(=O)NCCN(C(=O)CCN2CCOCC2=O)C)CC1=O Cc1cccc(C(=O)NCC(C)(C)OCC(N2CC3=C(C2)CN3C)=O)c1F O=C1CC(C(N2CCCOC(CNC(=O)C=CC=C(Cl)Cl)C2)=O)CC(=O)N1 c1(N2CCC(C(CC)C)CC2)ccc(Br)c(S(=O)(=O)NC(C2(OC)CCC2)C)n1 c1(C(=O)NCC(CC(=O)NC2(C(N)=O)CCCOC2)OC)ccnc(C)c1N c1(N2CCC(C(=O)OC3CCOCC3)C2)ccc(NC(C2CCNC2)=O)cc1 S(=O)(=O)(c1ccccc1C#N)Nc1c(C(C)OC)cc(F)cc1 N1(C(CCCC#CC)=O)C2CCC1CC(N(C)C(C13CCC(OC)C1C3)=O)C2 CCC1CN(C2CCN(C(c3ccc(=O)n(C)c3)=O)CC2)Cc2ccccc21 N1(C(C=CC)=O)CCC2(CC1)CC2C(=O)N(C1CC1)CC O=C1CC(C(=O)NC2CCN(C(=O)Cc3cnc[nH]3)CC2)Cc2ccccc21 CC(C)CC(C)(O)C(=O)N1CCN(C)C(C(N2CCC2c2ccccc2)=O)C1 N1(C(CC(C)OC)=O)CCC(C)(C)C(NC(c2ccc(C)cc2Cl)=O)C1 N1(C(c2c(OC)nccn2)=O)C2CCC(C2)C1CC(=O)NC1(c2ccsc2)CC1 N1(C(C(CC#C)NC(=O)CNC(=O)OC)=O)CCC(O)CC12CC2 CC1CCCC=C1C(=O)NC(C)(C)CCNC(c1conc1C1CCCO1)=O C1(CNC(CCCSC)=O)CCN(C(c2cnn(CC3CCC3)c2)=O)CC1C Cc1ccc(C(N2CCCC2CNC(C2CC2C2CC2C)=O)=O)cc1Cl C1(C(=O)NCC23CN(C(CC(=O)OCC)=O)C(C2)CO3)CCCCC1C1CC1 c1(CNCC(Cn2cc(COCc3ccccc3)nn2)OC)cnc(SC)nc1 C(=O)(C(C(C)NC(c1cn(C)nc1OC)=O)C(C)C)NC(CCCC)CCC C(CC(C(=O)N1CC(O)(C#N)C1)NC(=O)Cc1cnn(C)c1)SC CC(O)C(C(=O)NCCCNC(C12CC1C2)=O)N(C)C.c1(C)ccoc1 c1(C(N2CCC(O)(CF)CC2)=O)cc(-c2cc(F)ncc2F)cc2c[nH]nc12 c1(OC)ccc(C(N2CCCC2C(=O)N(C)Cc2ccccc2)=O)c(Br)n1 c1(CC)c(C(=O)NCC(C2(O)CCN(C(=O)CN(C)C(N)=O)C2)C)csc1C C(C(=O)NC(C)C(CO)NC(=O)C(O)CC1CCCCC1)(C(C)C)OC C(C)(CCC(=O)N1CCC(CCNC(=O)CCCF)C1)SC C(CCC(F)(F)F)ONC(=O)C1(N(C(C(=Cc2ccccc2)C)=O)C)CC1 C1(NC(CC(CNC(CCNC(C)=O)=O)OC)=O)CCC(C2CC2)C1 N1(CC(N2CCC(CN(C(=O)CSC(F)F)C)C2)=O)CCCC(C(N)=O)C1 c1(C(N(C)Cc2ccc(Cl)cc2Cl)=O)c(Cl)nc(Cl)c(Br)c1Cl C#CCC(C)(C)NC(=O)CC1CCCC1NC(=O)CSCCCN(C)C CC(CC(=O)NCC1CC(NC(c2cnc3nccn3c2)=O)C1(C)C)P(C)(C)=O N1(C(C2C(C)(NC(c3cnc(C4CC4)nc3)=O)CCCC2)=O)CCC2CCC(C2)C1 c1(C=O)nnn(C)c1CC.C1(C(=O)N)C=CC(C(=O)NCC2CC(OCC)C2)C1 CC1OC2(C(N3CC(O)(C(C)NC(=O)CCCC4CC4)C3)=O)CC1C2 c12ccc(c(OC)c1)CN2c1ncnn2cccc12.C1(CO)(CC2CC2)COC1.CO CN(C)S(=O)(=O)N(C)CC(=O)NCCC1(O)CN(C(C2CC(CF)C2)=O)C1 c1(NC(C2N(Cc3c(C)cccc3)CCNC2)=O)c(C)ccc2ncccc12 Cc1cc(C(=O)NC23CCCC2N(C(=O)CC2CC24CC4)CC3)cc(C)c1Br N1(C(C2CCC2CO)=O)CCC2CC12CC(N1CCC(C(F)F)C1)=O CCCCC(C)C(=O)NC1(C)CCN(C(C2CC3(CC3)C2)=O)CC1 c1(C(=O)NC(CN(C(c2c(CC)nco2)=O)C)CC)cnn(C)c(=O)c1 c1(C(=O)NC(C2CCN(C(CCN(C)CC)=O)CC2)C)cc(Cl)c(O)c(Cl)c1 c1(CC(N2C3CC(CNC(C(CSC)OC)=O)C2CC3)=O)ccc(F)c(Cl)c1F C(=O)(CC(F)(F)F)NC(CCNC(C(C1CCC(=O)N1C)C)=O)(C)C c1(CN2CCN(CC3CCCN(C(C)=O)C3)CC2)cnn2c(Br)cccc12 c1(C(=O)O)ccc(Cl)cc1F.c12ccc(F)c(c1)C(=O)NN1C(C)(CC1)C2 n1(CC)cnc2nc(N(C)Cc3ccccc3C#N)[nH]c(=NC3CN(CC)C3)c12 C(=O)(C1=CC2(CCN(C(=O)C=CC(F)(F)F)C2)C1)N1CC(C)(C)C1 c1(C(=O)NCC(CNC(c2c(OC)nccc2)=O)O)cnc(C)c(N)c1 C1(NC(C(CC=C)NC(c2cc(C)[nH]n2)=O)=O)CCCC(O)CC1 c1(NC(CCc2c(OC)ncc(Br)c2)=O)ccc2c(C)cc(Cl)nc2c1 C1(C#N)(C(N2CCC(O)(CN(C(CCOC(C)C)=O)C)C2)=O)CC2CC2C1 Cn1ncc(C(=O)NCC(C)(C2CC2)NC(=O)CC2(C)CC2)c1C#N C1(NC(=O)CSC2CC2)CCCCCN(C(=O)C(O)CC(F)(F)F)C1 N1(c2cc(OCC)ncn2)CCC(O)(C2(NC(=O)C(C)(CC)OC)CC2)CC1 O=C(C1=C(Cl)CCC1)N1CC(C(=O)NCC2CC(=C3CCC3)C2)CC1CO c1(C(N2CCN(C(c3nc(C)sc3)=O)C2(C)CCO)=O)ccc2ccnn2c1 C(C(CNC(=O)COCC(C)(C)C)C(F)(F)F)NC(c1cc(C)oc1C)=O c1(C(N2CCC(NC(C3C(OCC)C3)=O)C2(C)C)=O)cccn2ccnc12 N1(C(CN(S(CC)(=O)=O)C)=O)CC(NC(c2cnn(CCO)c2)=O)C(C2CC2)C1 c1(C(=O)NCC2COCCN2C(=O)CCc2nc(O)n[nH]2)ccc2ncnn2c1 N1(C(C=CC=CC)=O)CCC(C(C)C(N2CCC(c3ncco3)C2)=O)C1 N1(C(C(C)OC2COC2)=O)CC2(CCC2)CC1CNC(=O)CCCCNC(N)=O C1(C(=O)NCCn2ncc(CC)c2)CC(O)CN1C(=O)C(C)n1cccc1 N1(C(CCN(C(C(=C)F)=O)C)=O)CCN(C)C(=O)C1C c1(N(C)C)nccc(C(=O)NCCNC(c2cnn3c2OCC3)=O)c1Br C1(NC(=O)Cn2ncnn2)COCCN(Cc2ccncn2)C1 c12cccc(n1)NC2=O.c1(N(CCCOC)C)ccccn1 C1(F)(CNC(C(c2n(C)cnc2)O)=O)CCC(CNC(=O)CC2(C)CCCC2)C1 C=C=CC(C)C(=O)N(C1CCN(C(=O)C(C)NC(=O)Cc2ccccc2)C1)CC C(=O)(CC(N)C(=O)O)NC(CC(C)C)CN(C)C C(=O)(C1=CCCC1(C)C)N1CCC(C(C)(C)NC(COc2cc(C)on2)=O)CC1 CCCC(O)C(=O)N(C)CCN1CCN(C(=O)CSCC(N)=O)CC1 C(=O)(C(C)(C)C(F)F)N1CC(C=C)(CC(=O)N(C)CCN(C)CCO)C1 CC(C)CC(C)(C)NC(C1CCC1CNC(=O)CC1OCCC1(C)C)=O C(=O)(C(C)(C)C(F)F)NC(C)C(C)C(=O)N(C)Cc1ccco1 C(C(=O)NCCCCC1CN(C(C2CCCC(C)C2)=O)C1)(C(C)C)NC(C)=O C1(NC(CCN(S(C)(=O)=O)C)=O)CCC(N(C(=O)CC2CC(C)(C)CO2)C)CC1 C=C(Cl)CCC(=O)NCC1CN(C(c2cnc(N(C)C)cn2)=O)CCO1 C1(NC(CCN(CCCO)C(C2C(C)CC2)=O)=O)CCN2CCCC12 CC1CCn2c(C(N3CCCC(NC(=O)CCC4CC4)C3)=O)cnc2C1 C(C(CC)N=c1[nH]c(=NC)[nH]c(=NCc2cc(C)nc(C)n2)[nH]1)CCN(CC)CC CC1CCCN(C(C2CCC(C)(F)CC2)=O)C1CNC(C12CCCC(CO1)C2)=O CC1CN(C(=O)C(C)(C)c2cncs2)CC1NC(c1cnco1)=O C1(C(=O)NC)COCCN(Cc2cccc(F)c2Cl)C1.C12CCC(CC1)C(=O)N2 C1(C(=O)NCCc2nc(C)oc2C)CC(C)(C)CN1C(=O)C(C)Cn1ccnc1 N1(C(CN(C)C)=O)CC(CNC(c2nsc3ccccc23)=O)OC(C)(C)C1 c1(CC(=O)NC2CCCC(NC(c3c(C)cn(C)c3)=O)C2)ccc(F)cc1F n1(C(C)C)ncc2cc(C(=O)N(CC(C)NC(c3cnsn3)=O)C)cnc12 C1(CCNC(c2ncc(OCC)nc2)=O)CC2CCC(C1)N2C(=O)C(CC)CO c1(C(NNC(=O)C2CCCCCC2)=O)cc2c(cc1[N+](=O)[O-])OCCO2 C(=O)(C(F)(F)CCn1ccnn1)NCC(CNC(CSC)=O)CO c1(C(=O)NCC(CNC(c2c(C)ncn2C)=O)C)cc([N+](=O)[O-])ccc1N c1(C(=O)NC2(C)CCN(C(C3COCCOC3)=O)C2)ccc(F)c(F)c1 c1(N2C(CNC(C3C(C)OC(C)C3)=O)CCCC2)ncnc2sccc12 CCC(C)(CN=c1cccc(S(=O)(=O)N(C)Cc2cc(C)cs2)[nH]1)C(N)=O C(O)(C(F)(F)F)C1(C(=O)NCCOC2CN(C(CC3C(OC)CC3)=O)C2)CCC1 c1(CC(=O)NC(CN(C(=O)CCCc2nc(C)cs2)CC)C)ncn(C)c1C Cc1cc(C)c(C(=O)NCCC(C)(C)NC(=O)CC2CC2(C)C)c(C)c1Br c1(CC(N2CC(NCN(C(C3(OC(C)=O)CCC3)=O)C)C2)=O)cc(O)ccc1C CC1CN(C(c2cscn2)=O)CCC1C(=O)N(C)CCC1CCCC1 C#Cc1ccc(F)cc1C(=O)NCC(C1CC1)NC(c1c(F)cc(Cl)cc1F)=O N1(C(c2nc(OCC)oc2)=O)CC(NC(=O)C(C(C)C)NC(=O)COC)C(C)C1 c1(C(N2CC(CCNC(C3CC(CF)C3)=O)C2)=O)ccnnc1 c1(C(=O)NC2CN(C(CP(C)(C)=O)=O)C2)ccc(Br)c(F)c1N c1(OC)c(C(=O)NC2C3CC2N(C(c2ccnc(C)c2)=O)C3)oc2ccccc12 C1(C(=O)NC2CC(NC(=O)Cc3cc(C)no3)C2)(CC)CCOC1 C1(OC)CN(C(=O)COc2ccccc2Cl)CC1NC(=O)C(N1CCSCC1)C c1(C(N(CCCNC(c2c(C)snc2)=O)C(C)C)=O)cc[nH]c(=N)c1Cl O=C1NCc2c1ccnc2C(N1CCCN2CCCC2C1)=O N1(C(Cc2scc(C)c2)=O)CCC(F)(C(=O)NC(c2ncn(C)n2)C)CC1 c1(C(N(CC(CN(C(c2cnc(C(C)C)s2)=O)C)O)C)=O)ccc(F)nc1 c1(CN(C(=O)C=CCN(C)C(c2ccsc2)=O)C)ccncc1 C1(N(C(CC(=O)NC)=O)CC)CCCN(C(c2nc(C)oc2C)=O)CC1 C1(NC(CNC(c2nn(C)c(Cl)c2)=O)=O)CC2CCC(C1)N2CC1CCCCC1 N1(CC=CC(=O)NC2CC(CNC(C=CC(C)C)=O)C2)CCOCC1 N1(C(C(CCC)=CCC)=O)CCC(NC(C23CCC(C2)OC3C)=O)C(CO)C1 C(CCCC(CO)NC(=O)Cc1coc(C)n1)NC(C1CN(CCC)C(=O)C1)=O C(=O)(CCCCC(=O)NOC(C)(C)C)N(CCNC(c1c(C)coc1)=O)C CC1CCN(C(C2(F)CCOCC2)=O)C1CNC(=O)CSCc1ccccn1 N1(C(Cc2ccc(C)nc2)=O)CCCC(O)(CNC(=O)C2=CCCCC2)CC1 C=CC(C)(O)CC(=O)N(CC(C)(C)C(=O)N1CCC1COC)C N1(C(C2(F)CCOCC2)=O)CCC2(NC(C3CN(C(=O)NCC)C3)=O)CCCC12 C(C(CC(C)C)NC(c1[nH]nnc1C)=O)NC(c1cnc(C)s1)=O C(CC(C)(C)C(=O)N1CC(NC(C2CC(=O)N2)=O)C(n2ccnn2)C1)OC n1(C(C)C)cnc(C(N2CC(C)(NC(=O)Cc3ccn(C)n3)C2)=O)c1 C12(CCCOC1)C(=O)NCCCC2.C(C)(C(=O)NCCOCC)OCC=C Cc1nc(C)n(CC(=O)N(C)CC2CN(C(c3nnc(S)n3C)=O)C2)n1 CC(C)CC(CC(=O)NCCC1CCC(C)(C)O1)NC(c1ccc(CO)s1)=O N1(C(c2cc(C)n(CCO)n2)=O)CCN(C(=O)CC2CCC(O)C2)C(CO)C1 C1(NC(CCCN(C(C)=O)C)=O)CC(C)N(C(=O)CN(C(=O)C(C)C)C)C1 CN1CCN(CCC(=O)N(C)CC2(O)CCN(C(=O)CC3(C)CC3)C2)CC1 c1(N2CC(C(C)(C)NC(CCc3ccc(SC)cc3)=O)C2)ncc2sccc2n1 C(=O)(C(F)(CNC(c1sc(F)cc1C)=O)C(C)C)NCC(C#C)OC C1(C)(NC(CC2(C(=O)OC)CC2)=O)CCCN(C(C2CCC(C(N)=O)N2C)=O)C1 c1(C(N(CCCNC(CC=C)=O)C2CC2)=O)cc2c(cnn2C)nc1C CC1CN(C(c2cn[nH]c2)=O)CC1CNC(c1c[nH]nc1C1CCC1)=O NC(=O)CCCC(=O)NC1CC(CNC(=O)CSCc2ncc[nH]2)C1 C=C1CCN(C(c2cccnc2S)=O)C(C(N2CC(=O)NC(C(C)C)C2)=O)C1 C1(C(N(C2CCC(NC(C3CC(=O)C3(C)C)=O)CC2)C)=O)CCCCN1N=O c1(C(=O)NCC2CCN(C(C)C)C2)cc[nH]c2nccc1-2.C(C(F)(F)F)O N1(c2nnc(C)o2)CCC2(COC(CNC(=O)Cc3cn(C)nn3)C2)C1 c1(C(C(=O)NCCNC(c2ccc(OC)cc2)=O)=O)ccc(Cl)cc1OC c1(OC)ccc(-c2ccc(C(N3CCCCC3C)=O)cc2)cc1C=O.OC N1(C(C(C=CC)O)=O)CCC(CNC(c2c(C)cccc2OC)=O)C(F)(F)CC1 C1(C(=O)NC(CC)(C)C)CCOCCC1C(F)(F)F Cc1csc2c(C(N3CCC4(CC3)CC4CNC(C3(C)CC3)=O)=O)ncnc12 c1(CNC(C2OCCN(Cc3c(C)ccc(Br)c3)C2)=O)cnc2ccccc2c1 C1(C(=O)NCCCC(C)NC(c2ccnc(Cl)c2F)=O)CCCC12CCC2 c1(C2(c3ccccc3)C(C(=O)Cn3cc(-c4ccsc4)nn3)C2)ccc(Cl)cc1 C(=O)(CCCCCCNC(=O)C1=CCCCCC1)NC(CCC)C1CC1 c1(C(N2CC3C(NC(CS(CC)=O)=O)(C3)C2)=O)c(C)nn(C)c1Br c1(CC)ccccc1-n1nc(CC)nc1COC(C)C(=O)Oc1c(OC)cccc1 C1(NC(c2ccc(Cl)s2)=O)CCOC(C(N2CCC(O)C2)=O)C1 Cc1[nH]nc(C(N2CCC(C(=O)N(CC(F)F)C3CCC3)C2C)=O)c1C CCC(C)C(O)C(=O)NCCCCCCNC(C1COCC1(C)C)=O c1(OC)cccc(F)c1C(=O)NC1CN(C(=O)Cn2ncnn2)CCC1C N1(C(c2c(Br)cn(C)n2)=O)CCCC(C(N2CC3CCC2C3)=O)CC1 C1(CN(C(C2(c3cn(C(C)C(=O)OC)nn3)CC2)=O)C)COc2ccccc2O1 C1(CC=C)(NC(=O)CC2(C)CN(C(c3cncn3C)=O)C2)CCCC1 c1(N2CCC(C3(C)CC3)C2)nc2c(c(=NCCc3cc(Br)no3)[nH]1)CSC2 c1(CCC(=O)N(C(CNC(CC(CC)C)=O)C)C)ccc(N)c(F)c1 N1(C(Cc2ncc(C(=O)OC)[nH]2)=O)CC2C(N(C(=O)C(C)CO)C)C2C1 CC1(CC(N2CCCC(C)(F)C2)=O)Oc2ccccc2NC1=O C=C1CCC(CNC(=O)CNC(c2c(SCC3CCC4CC34)nc[nH]2)=O)CC1 Cc1cc(C(c2nnnn2CC2CC2)NC(CC)C2CC2)cs1 Cc1ccc(Br)cc1C(N1CC2CC(NC(c3ccco3)=O)C2C1)=O c1(NC(CC2CCC(NC(=O)OC)C2)=O)cc(C(=O)NCC(=O)N(C)C)nn1C c1(C(=O)NCCC(C)NC(C(CSC)O)=O)cccc(C(=O)N(C)C)c1 N1(C(CCN2CCN(C)CC2)=O)CCC2CN(C(c3cccc(N)c3O)=O)CC12 CCC(CC)(C(=O)OC(C)(C)C)C(=O)NC1CCCC1OC C1(NC(c2c(C)nc(C3CC3)o2)=O)CCN(C(c2ocnc2C)=O)C(C)C1 CC(C)CCC(=O)C(=O)N1CCC(C(F)C(N2CC(O)C(O)C2)=O)C1 C1(CNC(=O)C=CC=CC=C(Cl)Cl)(OC)CCN(C(c2ccon2)=O)C1 C1(COC(C(=O)NCCC(OC)OC)=O)Cc2cc(Cl)ccc2O1 C=CCCCCCC(=O)N1CC(C)(C(=O)Nc2cc(C)c(O)c(C)c2)C1 N1(C(CC(=C)C)=O)CC(C)N(C(c2c(F)ccc(F)c2OC)=O)CC1C N1(C(C2CC23CCCC3)=O)CC2CCCCCC12 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCC(C2CC2)(CNC(=O)CNC=O)C1 C1(C(=O)NCC(CN(C)C)O)CCN(C(=O)CN2CC=CC2)C(C)(C)C1 c1(OC)ccc(C)nc1C(=O)NC1CCC12CN(C(c1ccc(F)cc1N)=O)C2 CCCC(C(=O)NC)NC(=O)C(=O)NCCc1cccn1C C(=O)(CC(C)C(F)(F)F)N.C1(C)(CN(C)CC)CCN(C(C2CC(CF)C2)=O)C1 C(C)(C)(CC(C)(c1nnnn1CCC(=O)OC)NC(c1nc[nH]n1)C)OC c1(C(N2CCCC2CCCNC(C2(CC3CC3)CCC2)=O)=O)ccn(C(F)(F)F)n1 N1(C(C=C(C)C)=O)CC(NC(=O)CC2CCC(C)C2)C(n2cccn2)C1 CC(C)(C)C#CC(=O)NC1CCC(NC(c2cc3occc3[nH]2)=O)C1 c1(C(=O)OC)cnc(F)cc1C(C)(C)NCCc1cocn1 Cc1nc2ccccc2n1CCCCNc1cc(NCC(F)CO)ncn1 CC(C)C1=NOC(C)(C(=O)NCC23CC2CN(C(=O)C(c2ccccc2)=O)C3)C1 c1(NC(=O)NCC2CCNCC2)nc2ccccn2n1 c1(C(=O)O)ccc(S(=O)(=O)CCN2CCC(c3ncco3)CC2)cc1 C1(C#N)(OC(C)(C(=O)OCCN(C(C)(C)C)C)C2CCC2)CC12CCOCC2 C1(C(=O)NCC2(C)N(C(C(C(COC)C)C)=O)CCC2)CC12CCS(=O)(=O)CC2 N1(C(C(COC)N(C)C)=O)CC2CC1CN2C(c1ccnc(C(F)(F)F)c1N)=O C(CCSCC1(c2nnnn2CCCF)CCC1)(C(F)(F)F)OCC.C(C)(C)(C)O C(C(C)C(=O)N(C(C)CNC(=O)CNC(c1ccccc1)=O)C)OCC c1(C(N2CCC(O)(CNC(C3(O)CC(C)(C)C3)=O)C2)=O)ccn(CCO)c(=O)c1 c1(C(=O)NC(CC(C)NC(c2c(C)c[nH]n2)=O)C)cc2ccc(Cl)cc2s1 N1(C(C(C)NC(CC)(C)C)=O)CCC(F)(CNC(c2ccoc2)=O)C1 c1(OC(C(C2Cc3nnsc3S2)CCC)=O)cc(=O)oc2c(C)cc(C)cc12 N1(c2cc(NCc3[nH]cnc3C)nc(C)n2)CCC2(CCC2)S(=O)(=O)CC1 C1(NC(C=CC)=O)CCOC12CCN(C(=O)C(C(C)C)c1cnc(C)s1)CC2 Cn1ccc(=O)c(C(=O)NC(c2ccc(F)cc2)CNC(C2OCCO2)=O)c1 C=C(C)CC(C(=O)NCC1CN(C(=O)CC2(O)CCCC2)CCN1C)OC c1(C(N2CC3(CN(Cc4c(OC)cccc4OC)C3)C2)=O)nc(C)c(C)nc1C c1(CCNC(c2ccc(C)cc2C)c2n(CCCC)nnn2)cccc(F)c1F S(=O)(=O)(c1ccc(NCCC(N2CCOC(C)C2)C)c(Cl)c1)NC(CCC=C)C c1(C(N2C(C)CC(NC(c3cc(C4(C)CC4)on3)=O)C2)=O)cccc2nccn12 C12(CNC(=O)CC3CCSC3)CCC(NC(c3ccnnc3O)=O)(CO1)C2 c1(C(=O)NC2CC(NC(c3cocc3Br)=O)C2)ccncc1Cl C1(C(=O)NC(CC)CCCC)CCCN(C(c2cnn(C)c(=O)c2)=O)C1C CN1C(=O)OCC1C(N1CCCC(CNC(C2(C3CCCCO3)CCC2)=O)C1)=O c1(C(=O)NC(CCCC)CNC(C2(C(=O)N(C)C)CC2)=O)cc(C)ccc1Cl Cc1cc(CC(=O)NC2CC2CNC(=O)COC2CCCCCC2)c(C)s1 CC(C)(C)C(CNC(c1ccoc1)=O)C(=O)NCCCCSC(F)F CC(=O)CCN=C(NCc1cc2c(s1)CCCC2)N1CCC(n2cc(C)cn2)C1 C1(C(=O)NCC2C(C)CCN2C(c2cnc(O)s2)=O)CCC2(CC1)CC2 C#Cc1ccc(F)c(C(=O)NCC2CN(C(=O)CCCc3cncs3)CCO2)c1 N1(C(Cc2cc(COC)on2)=O)CC(NC(C23CC(C2)S(=O)(=O)C3)=O)CC(C)C1 c1(-c2onc(Cn3c(C)csc3=O)n2)c(F)cc(F)cc1F N#Cc1ccc(N)c(C(=O)NCC2CN(C(=O)C3CC3)CCC2C(F)(F)F)c1 Cc1nc(C(F)(F)F)c(C(N2CCC=C(Cl)C2)c2nnnn2C2COC2)s1 c1(C(=O)NCC2(F)CCN(C(C3(F)CC=CC3)=O)C2)ccc2c(c1)CCC2 CCN(OC)C(=O)CCNC(=O)CCc1cncn1C C1(CC=C)(C(=O)NCC(CC2CC2)OC)CCCN1C(c1cc(CC)n(C)n1)=O N1(C(Cc2n(C)nc(C3CC3)c2)=O)CC(CNC(C2CC2CF)=O)CC(C)(C)C1 N1(C(c2ccc(CC)nc2)=O)C2CCC1C(C(=O)Nc1cnc(OC)c(C)c1)C2 C(=O)(CC(C1CC1)NC(C)=O)NC(C(=O)NC(CC)C)C1CCCC1 N1(C(C(C)=CC)=O)CCCN(C(=O)C(C(C)C)c2cnn(C)c2)CC1 CCC(F)C(=O)NCCOCCN(C(=O)C(C)OC1CCCCC1)C c1(NC(c2cc(Br)c(C)o2)c2n(CC(=C)C)nnn2)cccc(CO)c1 CCCCCCCC(=O)N1CCC2(CC2C(=O)Nc2ccc(I)cc2C#N)C1 c1(C(N2CCCC(NC(c3nccc(C)c3)=O)CC2)=O)cc2nc(C)ccc2o1 C1(c2nnnn2CSc2ccccc2)(NCCCNS(C)(=O)=O)CC2CC1CC2 N1(C(c2ncn(C(C)C)c2)=O)CCC12CN(C(=O)C=Cc1ccncn1)C2 C=CC1(C2(C(N3CCC(NC(=O)C(F)(F)CC)C(F)C3)=O)CCC2)CCC1 C1(CNC(COCCOCC)=O)CC2CCC(C1)N2C(=O)CCc1ccc(C)s1 c1(CC(C(=O)N(C(=O)CN(C(C)S(=O)(=O)C(C)C)C)C)C)ccc(O)cc1.CO C1(CC)CCCC1C(=O)NCCCN(C(=O)CCN1CCCC1=O)C N1(C(C2(C=C)CCCCC2)=O)CC(NC(C2(F)CCOC2)=O)C(C2CC2)C1 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C)CN(C(=O)CCSc1nnnn1C)C CC1CCn2cc(C(N3CC4(CCN(C(=O)C(C)(C)CCCO)C4)C3)=O)nc2C1 C(=O)(C1CCc2cccnc21)NCC(CN(C(CCC(=O)NCC)=O)C)(C)C C(=O)(CCC(F)(F)C(F)F)N1CC(CNC(C2C(C)(C)C2)=O)OC2C1COC2 CC(C)CCC(O)C(=O)NC1(C(=O)NOCC2CCCO2)CCOCC1 N1(C(CC)=O)CC(CNC(=O)CSc2nc3ccccc3[nH]2)N2CCC1C2 C1(CNC(c2cnc(C(C)=O)s2)=O)CCCN(C(=O)C(Cl)=CCl)C1 C(=O)(C(c1ccoc1)NC(=O)C=CCO)NC(C)CN(C)C CC1CC2(CCC2)CN1CCCOc1cccc(C(=O)O)c1 C(=O)(CCCCc1ccccc1)NC1CC(N(C(=O)CC2(O)CCCC2)C)C1 Cc1cc(C(=O)NC2CC2c2cccc(Cl)c2)ccc1C#N c1(NCCc2ccc(Cl)c(Cl)c2)nccc(=NC2CC3(CCC3)C2)[nH]1 N1(C(c2cnc(C)[nH]2)=O)CCCN(C(c2cc(-c3ccoc3)[nH]n2)=O)CC1C c1(C(=O)NCCCC)ccc(C(c2csc(Br)n2)c2nnnn2CCCF)cc1 CC(O)C(F)(F)C(=O)NCCC1CN(C(=O)C(F)=C2CCCC2)CCO1 C1(C(=O)NC(C)C(CO)NC(C2(C)CCCCCC2)=O)CC12CCCCC2 C1(NC(C2(C)CCOC2)=O)CCCCC1CC(=O)NC.N1(C(C)(C)C2CC2)CCOCC1 Cc1cc(N2CC(NC(c3cccnc3CO)=O)C(C)(C)C2)nc(C)n1 C(=O)(C#CC1CCOCC1)N1CC(CCCNC(CSCC(C)C)=O)OCC1 c1(C(=O)NC2CC(C)N(C(=O)C(=O)NC(C)(C)C)CC2)cnc2c(c1)CCCO2 c1(C(N2CCN(C(Cc3onc(C)n3)=O)CC2CO)=O)c[nH]c2cc(Cl)ccc12 Cc1nccc(C(=O)NC(c2ccccc2)CC(C2(C(=O)C3CC3)CC2)=O)n1 C(=O)(C(C)(C(C)C)OC)NC1C(OC)CN(C(c2ccnc(C)c2)=O)C1 CC1(C)CN(C2C(O)C3CCCC23)CC(C)(C)O1 C(=O)(CCC(=O)NN(C)C)NCC(CN(C(c1c(C)cc(O)c(Cl)c1)=O)C)(C)C CN1CC(C(=O)NC2CCCC2NC(=O)C(F)CC2CCOCC2)CCC1=O C1(N(c2c(CN(C)C(=O)NCc3ccccc3)cccc2)C)CCCCC1(C)O CCCC(C(=O)N(C1CN(C(=O)CC2=NNC(=O)C2)C1)C)S(N)(=O)=O C(=O)(C(C)(F)C(=O)N1CCC(F)(C(=O)NC(CO)CC(F)(F)F)CC1)OC S(=O)(=O)(c1cccc(=NC(C)C2CCCO2)[nH]1)NCC1(C(=O)NCC)CC1 n1(CC2CCN(C(C(F)OCCC3CN(CC)C3)=O)CC2)cnc2ccccc12 C=CCCCC(C)(C)C(=O)NC1CCC(F)(CNC(=O)Cc2cnco2)C1 C1(CNC(CC(CC)C)=O)CN(C(C2CC2(C)C)=O)CC2(CCC2)O1 C(C1CN(c2ccc([N+](=O)[O-])cc2)Cc2ccccc21)NC(C1(C)CC1(F)Cl)=O N1(C(C(CC)N(C)C)=O)C2CCC1C(F)C(NC(c1cn3ccsc3n1)=O)C2 Cc1ccccc1C(N1CCCCC1c1n[nH]cc1C(=O)NC1CCOC1C)=O N1(C(C2ON=C(C)C2)=O)CCCC12CCN(C(c1cc3n(n1)CCC3)=O)C2 C1(NC(CS(=O)(=O)N(C)C)=O)CCCCC12CCCN(C(=O)Cc1ccoc1)C2 c1(C(=O)NC(c2c(SC)cccc2)C)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] c1(C(N2CC(CNC(CCC)=O)C(C)(C)C2)=O)c(C)nc2sc(C)cn12 C(C(CCO)CC(C)C)NC(c1cn(CCCCC(=O)OC)nn1)(C)C c1(C(N(C)CC2(CNC(=O)CC3CCOC3)CC2)=O)c(F)ccc(F)c1Cl Cc1c(Br)ccc(C(=O)NC2CC2C(=O)NCc2cccc3occc23)c1F N1(C(C2CCC(OC)CC2)=O)CC(C2CC2)(C(=O)NCCN2CC3CC3C2)C1 n1(CC)cc(C2OCCC2OC(=O)COCc2cccnc2)cn1 C1(C(=O)NC2C(CNC(c3ccc(CO)s3)=O)C2)CCCN(c2nccs2)C1 N1(C(c2on(C)c(=O)c2)=O)CCC2(CCCC2NC(=O)C2=CCCCC2)C1 N1(C(COCC(C)C)=O)CCN(C(c2ccc(-n3ccnn3)cc2)=O)CC1C c1(C(N(CCC(=O)N(C)Cc2cnco2)CC#C)=O)c[nH]c2ncccc12 c1(OC)ccc(F)c(C(N2CC(NC(c3cccc(Cl)c3O)=O)C(O)C2)=O)c1 C1(NC(C=CCNC(CC2C(=O)NC(=N)S2)=O)=O)CCOCC12CCC2 c1(C(=O)NCC2C(CNC(CSCCCC)=O)C2)cnc(C2CC2)cn1 N1(C(C2N(C(C(C)NC(CC)(C)C)=O)CCCC2)=O)CCC2CC1C(=O)N2C N12CCC3(CC1)CN(C3)C(=O)C1(CC1C)C2=O.Cc1oncc1C(=O)O C(=O)N1CCCO1.CC1(NC=O)CN(C(=O)CC23CCCC2C3)C1 C1(CSNC(C=CC)=O)CCCC12CCN(C(=O)Cn1ccc3ccccc13)CC2 C1(O)(CNC(C2C3CCCC23)=O)CCN(C(c2ccc(C(F)F)cc2)=O)CC1 Cc1ccc(F)cc1C(=O)C(=O)NCCC(C)N(C)C(c1cc(Cl)n(C)n1)=O C(=O)(C1=CCCOCC1)N1CC(C2CC2)(C(N(C(C#C)C2CCC2)C)=O)C1 c1(C(=O)NCC2CCCCN2C(C2C(C)C2)=O)cc2sc(=O)n(C)c2s1 c1(C(=O)NCCC2CC(NC(CN(c3ccccc3)CC)=O)C2)cc(C)c[nH]1 C1(CCNC(c2c(CC)noc2C)=O)CCCN(C(c2ccc(C#N)s2)=O)CC1 c1(C(=O)NC2(COC)CN(C(C3COCCC3C)=O)C2)nn(C)cc1S(C)(=O)=O Cc1cc(-n2cncn2)ccc1C(N1CCC2CCC12CNC(C1CSC1)=O)=O CCC(C)(COC)C(=O)NCc1ccc(C(=O)NC2(C)CC2)o1 C(=O)(C(COCC)N=[N+]=[N-])N1CC(C(=O)NC(CC)C(C)CN(C)C)(N)C1 C12(NC(C3C(C)C3)=O)CC1CN(C(C1(C)CCSCC1)=O)C2 N1(C(C2CC(CC)C2)=O)CCCC1CNC(=O)Cn1cnc(C(N)=O)n1 c1(CCC)nnsc1C(=O)NCC1CC(F)(CNC(=O)Cc2ccsc2)C1 c1(N(CC(=O)N(CCNC(C(C=CC)O)=O)C(C)C)C)ccc(C)c(CSC)c1 C1(c2n(CC=C)nnn2)(NCCc2ccc(C(F)F)cc2)CCN2CCCC12 N1(C(C=CC)=O)CC(NC(=O)C(C)CF)CC12CCOCC2 CC1CCC(C)N(C(C(=O)NCC2CC2)C2=CCCC2)C1 CC1CCN(C(=O)CO)CC1NC(c1nccn1C)=O C=CCC(CC)C(=O)N(CCCCC(=O)NC1CCCCNC1=O)C c1(C(=O)OC)ccc(C(=O)NCC(C)NC(=O)CCc2cncc(C)c2)c(C#N)c1 c1(NC(c2cccc(-c3cnn(C4CC4)c3)c2)=O)ccc(I)cc1I c1(C(N2CCN(C(C3=CC(C)(CC)C3)=O)CC2CF)=O)cnn2c(Cl)cccc12 C1(C(N(C2CC(O)C2)C)=O)CC1C1CN(C(c2ccnn2C)=O)C1 N1(C(C(C)OCC)=O)CC2CCN(C(C3CCCCCC3)=O)CC(C2)C1 C12CCCC(C1)C(=O)O2.c1(OCC(=O)NCCC(C)NC(N)=O)ccc(Cl)cc1 C1(C(=O)OCC)CCC1(C)C(=O)OCc1ccc(Cl)o1 N1(C(Cc2cc(OC)no2)=O)CCCC2CN(C(=O)CC3=CCCC3)CCCC12 c1(OC)ccc(CCC(=O)Nc2cc(Br)ccc2OCC)cc1O.C(C)(C)O N1(C(C(CO)N(C)C)=O)C(C(N2CCC2CC2CC2)=O)CCC12CC2 N1(C(C2(C(C)C)CC2)=O)CC2(CCCN(C(C3CC=CCO3)=O)C2)C1 C(=O)(C#CC1(C)CC1)N(CCC)CCN(c1cccc(Cl)c1)C c1(OC)cccc(C2=NOC(C(=O)NC(C)CNC(=O)C(C(C)O)N(C)C)C2)c1 C1(=O)C(C)C(C)N1.c1(CC(=O)NC2(C(=O)NCC#C)CC2)cnc(C)s1 N1(C(C=CC=CCC)=O)CCC(CNC(c2cc(N(C)C)ccc2F)=O)C(C)C1 C1(CNC(=O)NC(CCCC)CO)CC2CCCCC12 c1(C(N2CCC(N(C(C3CC(C)=NO3)=O)CC)CC2)=O)ccc2c(c1)NC(=O)C2 N(C(=NCCC1CCCCC1)NCCN1CCOCC1)C1C(N)CCCCC1 C#Cc1cccc(C(=O)NC23CC2CN(C(C2CC4(CCC4)C2)=O)C3)c1Cl C(C(C)C(C)C(=O)N1CCC(OCCNC(c2cccnc2)=O)CC1)OC CC(C)(C)CCC(=O)N1CCOC(CCCNC(=O)C=CC2CCOC2)C1 C#CCCC(C(=O)NC)NC(=O)CCCCNC(CO)CCSC C(=O)(N=c1cc(C)n(CCO)[nH]1)C1N(C(C(CCC)N(C)C)=O)CC=C1 c1(CC)nc(C=CC(=O)OC)cs1.C12CCC(CC1)C(=O)NC1CN(C1)C(=O)C2 C1(NC(COCC#C)=O)CCN(C(c2ccc(C(C)C)cc2)=O)CC1CC Cc1nn(C(C)C)c(C)c1C(N1CC(NC(=O)C(C)(C)O)CC(C)C1)=O N1(C(CSCCC)=O)CCC(CNC(C2(c3ccccc3)CC2(C)C)=O)CC1 N1(C(C(CCC)NC(N)=O)=O)CCC2CC1CN(C(=O)CCc1ccc(C)s1)C2 c1(-n2ncc(C(=O)OCC(=O)N(C3CCCO3)C)c2)ncc(Cl)cn1 N1(C(c2cn(CC)nn2)=O)CCC2CC1CN2C(=O)Cc1cccc2c1OCO2 Cc1c(C(=O)NC2C=CC(CC(=O)NCC3CCCCS3)C2)ccn1C N1(C(C2(CC)CC(F)(F)C2)=O)CCC(NC(C2(C3CCCO3)CC2)=O)C(C)C1 c1(C(C)(C)C)conc1C(=O)NCC(C)(C1CC1)NC(=O)C(C)(O)C1CCC1 C(=O)(C(O)CCS(C)=O)N1CCN(c2ncnc(N3CC=C(C)C3)c2C)CC1 O=C(C#CC1CCCCC1)NCC1N(C(=O)OC(C)(C)C)CCC1(F)F Nc1c(C(F)(F)F)nn(C2CC2)c1C(=O)NC1CCC1CNC(=O)Cn1ccnn1 c1(C(=O)NC(C2CCN(C(=O)CN3C(=O)CNC3=O)C2)C)ncc(Br)cc1N C(=O)(CS(=O)(=O)C1CC1)NC1CCCC(N(C(Cc2c(C)n[nH]c2C)=O)C)C1 C(C)(CCC(F)(F)F)NC(C1(CC=C)CCN(C(C2CC23CCCCC3)=O)C1)=O c1(OC)nc(C)ncc1C(=O)NCCCCC(C)NC(c1cccc(CO)c1)=O C=CC12CCN(C1)C2=O.C1(C(C)NC(=O)CN(C(C)CC)C)CCC1 N1(C(CCC(C)OC)=O)CCC(NC(C2CCCOC2)=O)C12CCC2 C(CC(C(C)C)NC(=O)CC1(N(C)C)CC1)NC(C(CC)SC)=O C1(NC(Cc2n[nH]c(=NC)s2)=O)CC2CC(NC(=O)CSC)C2C1 C1(C(c2scc(C)n2)=O)CN(C(=O)OC2COCCN2C=O)C2(CCC2)C1 C1(CNC(C2C(NC(CC3C(C)=NNC3=O)=O)CC2)=O)CCC(C)(C)CC1 c1(NC(=O)CC2CCCN2C(=O)CN2CCCC2)cc(C(F)(F)F)ccc1O c1(C(=O)NC(c2ccnn2C)C(=O)NC(CCC=C(C)C)C)ccnc(CO)c1 CC(O)CCCc1cn(CCN2CCC(C3C(C(=O)OC(C)(C)C)CC3)C2)nn1 C1(C(=O)NC2CC(F)(CNC(C=CC)=O)C2)CCn2c(C)cnc2C1 C(C(C(=O)NCc1cc(C)co1)C(C)(C)C)NC(C(COC(C)=O)C)=O c1(C(N(CCCNC(c2cn(C(F)F)cn2)=O)C(C)C)=O)nc(=O)n(C)[nH]1 C1(NC(c2ccc(CC)o2)=O)CN(C(C2CSCC(=O)N2)=O)Cc2ccnn2C1 N1(C(c2cnc(SC)nc2)=O)CC(NCc2ccc(Br)nc2)C2(CC2)C1 c1(C(N2C(CCNC(C3=NOC(C)(C)C3)=O)CCC2)=O)nc2ccccn2c1F C#CC1CCN(C(=O)CC2CCCN(C(=O)C(c3cccnc3)C)C2)C1 c1(C(=O)N=C2CC(C(=O)OCC)C2)ccc(C(N)=O)nc1.C12C(CC1O)NC2=O N1(C(C2CN(CC)C(=O)C2)=O)CC(N(C(=O)CSCC(F)F)C)C2(CC2)C1 c1(CCC(=O)NCCN(C(=O)CCOCC(C)(C)C)CC)nc(=N)[nH][nH]1 Cn1c(CCN=c2[nH]c(Cc3ccccc3)cs2)cc2ccccc12 CCC(C)CCCC(=O)NCCC1CSCCN1C(c1cc(CO)n(C)n1)=O c1(C(N2CCC(N(C)C(c3cc(C(N)=O)cs3)=O)C2)=O)cccc2c1COCC2 C(=O)(CCC(=O)NN(C)C)N1CC(CC)N(C(c2cc3c[nH]cnc-3n2)=O)CC1 C1(C)(C(=O)OC)CCCN(c2nn(Cc3ccc(Cl)cc3)cc2I)C1 Brc1ccc2nc(NC3CCN(CC)C3)[nH]c(=NCc3cc[nH]c(=N)c3)c2c1 CC(C)(CS(N)(=O)=O)NC(C12CC(NC(=O)CC3CCCC34CC4)(C1)C2)=O C1(CC)CCCC1C(=O)N(CCO)CCNC(=O)C=CC(C)(C)SC c1(C(=O)NCCOC2CN(C(C(C)C3CCCO3)=O)C2)cccc2sccc12 c1(CN2CCC(C3N(C(c4c(Cl)n[nH]c4C4CC4)=O)CCC3)C2)ccc(Br)cn1 c1(OC)cc(CCNC(=O)NCCNC(c2cn(C3CC3)nn2)=O)ccc1OC C(CCC(=O)NC(c1ccoc1)C)(C(C)C)NC(CCC#C)=O c1(N2CCC(C(C)NC(C3CC(C)OC3C)=O)C2)nc(Cl)nc(C2CC2)c1F N1(N2Cc3c(ccc(C=O)c3)CC2)CCc2cc(Br)cc(Cl)c2C1.CO CC1(CCC(=O)NC23CC(F)(C2)C3)CCCN1C(C1(C(=O)N(C)C)CC1)=O N1(C(C2CCC(SCC)CC2)=O)C2CCC1C1CC1(NC(=O)Cc1cnns1)C2 N1(C(CNC(COCCOC)=O)C)CCN(C(=O)CC2C=CCCC2)CC1 c1(CC(=O)N(CCCC(=O)Nc2ccc(O)cc2)C2CC2)ccc2c(c1)CC2 C1(C)(c2cn(C)nn2)CCNCC1.C1(COC)CC(COCc2ccccc2)NC1=O C=CCC(CC(C)C)C(=O)NC1CN(C(C2CCCC2C)=O)CC2(CCC2)C1 C1(NC(c2cc(CC(C)C)on2)=O)CCCC12CN(C(C1CCCO1)=O)C2 c1(CN(c2cccc(OCC)c2)CCC)cc(NC2CCNC2)ncn1 C1(C(=O)NC2CCCN(C(C3(C(C)C)CNC(=O)C3)=O)C2)CCC(C#N)CC1 c1(C(N2CC(NC(=O)C(F)(F)C(F)F)C3CCCC23)=O)cc(F)cc2ccoc12 C1(NC(c2ccnn2C(F)F)=O)CCCCN(C(=O)C=Cc2ccncc2)C1 N1(C(C2(C)CCCCC2)=O)CCC(NC(C2(c3cccc(Cl)n3)CC2)=O)C(O)C1 C(C)(C(C)NCC1(c2ccccc2)CCOC1)(C1CC1)NC(C)=O n1(CCSC)nnnc1C(c1ccccn1)NCC1(c2ccccc2)CC1(C)C C(=O)(C(F)(CC)C(=O)OC)NCC1(C(CC)=O)CC1.N12CC(C)(C1)OCC2=O C(=O)(C(CCOC)NC(c1cnsn1)=O)N(C)Cc1ccc(CC)o1 N1(C(CCSc2nc(C)[nH]n2)=O)CCCC2C1CCN2C(=O)C(C)(C)C1CCC1 c1(CC(=O)NC2CCC(NC(c3ccn(CC)c3C)=O)C2)c[nH]c2ccccc12 C(=O)(C(CC(C)(C)C)OC)NC1CC2CN(C(C(C)NC(CC)=O)=O)CC21 c1(C(N2CCC(CN(C(=O)COC3CCOC3)CC)CC2)=O)ccc(O)c(N)n1 c1(C(N(CCNC(C2CCC(=O)N2)=O)CC)=O)cc(C)n(-c2ccon2)c1C c1(C(C)C)ccc(N(C(=O)C(N2CCN(CCN)CC2)C)C)cc1 N(C(=NCCCC(C)(C)O)NCc1c(Cl)cccc1Cl)CC C(=O)(C1CC(O)c2ccccc21)NCC1C(CNC(c2cn[nH]c2)=O)C1 N1(C(C2CC(CC)OCC2)=O)CCN(C(c2ccc(Cl)c(O)c2)=O)C2(CC2)C1 CCC(CC)C(=O)N1CC2CC2(CNC(=O)CCC(=O)NC)C1 N1(C(C(=O)NC2COC2)C2CCSC2)CC2(CC2)CC1c1ccccc1 C(=O)(C(C)(C)CC(C)(C)C)NC1C(NC(c2nn(C)c(=O)cc2)=O)CCCC1 C1(C(=O)C(c2ccc(C)cc2Cl)C)CC(CC(N)=O)CCN1CC.CO C1(COC)CN(C(=O)COCC2CCOC2)CCN1C(c1ccc[nH]1)=O C(C(=O)N1CC2C(NC(=O)CCn3cc(Br)cn3)C2C1)(C(C)C)NC(C)=O C#CCCC(=O)NCCC1(C(=O)N(C)CCN2CCCCC2)CC1 C(=O)(CS(=O)(=O)N1CCN(C(=O)Cn2ncn(C)c2=O)CC1)OCC C1(C(N2CC(OC)C2)=O)CCCN(C(C2CC(F)(F)C2)=O)C1 C(=O)(C(C)CC(C)C(C)=O)NC(C(=O)N(C)Cc1scc(C)c1)CCF N1(C(C(CC)Cc2cccc(Br)c2)=O)CCN(Cc2ccccc2)CC1C C12(CNC(C(c3ccc(CC)s3)=O)=O)CC1CN(C(C1(C)CC=CC1)=O)C2 CC#CCC(C(=O)N(C)CCO)NC(c1cnc(CC)o1)=O c1(C(c2nnnn2C(C)C)NCCOCC=C)csc2cc(Cl)ccc12 C(=O)(CC(C)(C)CC(=O)N(CCC(N1CC(OC)C(C)(C)C1)=O)CCO)OC C(=O)(C(CC(C)C)NC(=O)C(O)c1ccsc1)NCc1cn(C(C)C)nc1 CC1(C)C(CNC(=O)CCc2cnco2)CCN1C(c1ncccc1O)=O C1(C(N2CCC(F)(CNC(CNS(CC)(=O)=O)=O)C2)=O)CC2(CCC2)CCO1 C1(C(=O)NCc2c(C)ccc(F)c2)CCN(C(c2cc(C)n(C)n2)=O)C12CCC2 C(N=C(NC1CC1C1CC1)NC1CC1)C1CC(Cl)C1 C1(NC(N(C2CCN(c3ccccn3)CC2)C)=O)CC2CC(N)C2C1 C1(C(N(C(C)(C)C2CC2)C)=O)CCC(CNC(=O)CSc2cnc[nH]2)CC1 CC(CC(=O)NCC1CN(C(c2ccccc2)=O)CC12CCC2)C(C)(C)C C1(CNC(CC(CC)C)=O)CN(C(=O)CCCCSC(F)F)CCC12CCOCC2 C(C(C)(C)C(=O)NCCC1COCCO1)NC(C(C)n1cccc1)=O C(C(C)(C)C)=CC(=O)NCCC1(CNC(COCCOC)=O)CC1 c1(N(C(=O)NC(C)CCc2ccc[nH]2)C)ccccc1 CC1CCCN1CCCN(CCCn1cc(-c2cnn(C)c2)nn1)C C(=O)(CCC(C)(C)N(C)C)N1CC(O)(C(C(=O)N(CCCC(C)(F)F)C)F)C1 C(=O)(C(CO)C(C)(C)C)N1CCC(C(=O)NCCc2onc(C)n2)C12CC2 C(C(F)C(=O)C1C2CCCC12)NC(NCC(=O)OC(C)(C)C)=S N1(C(C2C(=C)CC2)=O)CCCCC1c1cn(CC2CCCOC2)nn1 C=Cn1ncc(C(=O)NCc2nc(C(N3CCC(OC(C)C)C3)=O)c(C)o2)c1N CCCCC(C)CC(=O)N1CCC(Nc2ccc(C(C)(C)C)cc2)C(C)C1.C=O N1(C(C2C(C(C)C)OCC2)=O)CC2(CCN2C(=O)COc2cc(F)ccc2F)C1 c1(CNC(c2cnn(C)c2C(C)C)c2n(CCCSC)nnn2)cc(C)c(C)o1 c1(C(=O)NCC2(C(N)=O)CN(C(C3(SC)CCC3)=O)C2)cccn(C(F)F)c1=O C1(NC(c2c(C)nc(CNC(C3C(C)(C)CCO3)=O)o2)=O)CC(C)(C)OC1=O Cc1cnn(C(C)C(=O)NC2CC(C(C)NC(c3occc3C)=O)C2)c1 c1(CN(C)C(c2n[nH]cc2CNC(c2ncn(C)n2)=O)=O)nccn1C C1(CNC(c2cc(CO)[nH]n2)=O)CCCCN1C(=O)CCF c1(C(N(CCCC=C)C)=O)nc(CNC(c2ccc(O)nn2)=O)oc1C C(C)(CCC(=O)NC12CC(C1)N(C(=O)Cc1nocc1C)C2)n1ncc(C)c1 CC1CS(=O)CCN1C(c1nnnn1CCCF)(C)CN1CCCCC1=O N1(C(C(C(C)NC(C(CC)CCOC)=O)C)=O)CCC12CCC(C)CC2 c1(C(C2CCCCN2Cc2ccc(-c3nn[nH]n3)cn2)F)cccc(Cl)c1 C1(NC(C2CC(SC)C2)=O)CN(C(c2cc(C(F)F)nn2C)=O)CCC1C C(=O)(C1CCCc2nc[nH]c21)N1CC2(CC(CNC(C(F)=CC)=O)C2)C1 N1(C(c2cc(C#N)on2)=O)CCCC(NC(c2ccc(N3CCC3)cc2)=O)CC1 C1(CNC(c2nc(C#C)sc2)=O)CN(C(=O)CCN2CCCCCC2)CCC1C N1(C(C2(CCOC)CC2)=O)C2CCC1CN(C(=O)CCC1CC1)CC2 N1(C(Cc2c(C)n(C)nc2)=O)CCC2CC(CNC(C3CC3(Cl)Cl)=O)CCC2C1 N1(C(CC2N(C(C(C)NC=O)=O)C3C2CCC3)=O)CCCC12CCCC2O N1(C(C(CSC)O)=O)CCCCC(CNC(c2n[nH]cc2C2CCC2)=O)C1 c1(C(N2CCC(N(C(C(c3ccccc3)SC)=O)C)C2)=O)ccc(C#N)o1 O=C(C1=NOC2(CCC2)C1)NC12CCC1CN(C(c1ccc(O)c(Cl)n1)=O)C2 C1(C(N(C2CC(NC(C(N3C(C)CCC3)=O)=O)C2)C)=O)CCCCCC1 c1(C(=O)NCC(=C)CCNC(=O)CC2CC(F)C2)cnc(O)n(C)c1=O C1(CC(=O)NCC=C(C)C)CCCCN1C(=O)OCCl.C(C)(C)(C)O C1(CNC(c2coc(C(F)F)n2)=O)CC2CCCC(C1)N2C(=O)C(F)C1CCC1 N1(C(C2N(C(N)=O)CC(O)C2)=O)CCC2(C1)CN(C(c1cc(CO)ccn1)=O)C2 C1(NC(c2cnn(CC(F)F)c2)=O)CCN(C(C2CN(S(=O)(=O)C(F)F)C2)=O)C1 N1(C(C(c2ccccc2)OC)=O)CC2(CCC2)CCC1CNC(=O)C(Cl)=CCl C#CC12CCC(C(=O)NC3CCC(NC(C4CCC(CC)CC4)=O)C3)(CC1)CC2 CC1OCCC1C(=O)NCCCC1CCCN1C(=O)Cn1cnc(C(N)=O)n1 N1(Cc2c(N(C)C)cccc2)CCOc2c(Br)cccc2C1 C#Cc1ccccc1CNC(N1CCC(C(=O)OC(C)(C)C)C(C)C1)=O N1(C(c2sc(CC)nc2Br)C(=O)NCCCC)CC(C(F)(F)F)CCC1C N1(CCCN(C(=O)Cc2cnsc2)C)CCN(C(=O)Cn2cnccc2=O)CC1 C1(C(=O)NCC(C)OCC#C)(NC(c2cc(O)ncn2)=O)CCN(C)C1 C1(N(C(=O)NC2CC(C(C(=O)OCC)F)C2)C)CCc2nccn2C1 c1(C(=O)NCC(CC=C)NC(c2ccc(CO)s2)=O)ccc(O)c(F)c1F C(C)(C)(C(=O)N(CCCCCNC(C1(C(F)F)CCCC1)=O)C)NC(=O)OC c1(NC)ccc(S(=O)(=O)N2CCOCC2)cc1.C1(=O)CNC(=O)N(CC)CCN1 C(=O)(CCC(=O)NN(C)C)NC1CN(C(CC(C)c2ccncc2)=O)C1 c1(C(N2CC(CNC(c3c(CC)non3)=O)(COC)C2)=O)ncncc1Cl c1(NCC2(NC(=O)C3=CCC3)CCCCC2)ccnc2ncnn12 c1(CNC(C2CCC(CC(=O)NC3CCCO3)CC2)=O)cn2cccc(Br)c2n1 CCC(CC)(CC)C(=O)NC1CCC(CN(C)C(c2cc3n(n2)CCC3)=O)CC1 S(=O)(=O)(c1cn(C)cn1)N(C(C(C)C)C(=O)NCCCCNC(=O)CC(F)F)C c1(C(=O)NCC(CNC(C(C)(CO)OC)=O)O)ccc(F)c(Cl)c1 CCC(COC)C(=O)NCCCN(CCCCNC(C1CC1C(C)(F)F)=O)C CC1CN(C(=O)NC(C)(C)C)CC1n1cc(-c2cnccn2)nn1 c1(OC(C(=O)NC(C)CC2CN(C(c3ncc[nH]3)=O)C2)C)ccccc1Cl c1(C(N2CC(CCC)N(C(C3CC(O)C3)=O)CC2)=O)cc2sc(C)cc2s1 C1(C(=O)NC2CN3CCCC2C3)CC2(CC(=O)C2)C1.CC1OCCN2C1C2=O C(CCCCCCCC(=O)O)CN(C(C(N1CCN(C2=NCCS2)CC1)(C)C)=O)O N1(C(c2c(C)nc(COC)s2)=O)CC(NC(c2cnc(Cl)n2C)=O)CC(C)C1 N1(C(C(CCC)(C)O)=O)CCC2(CC1)CN(C(c1ccc(OC)nc1C)=O)C2 N1(C(COCCC=C)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1C1CC1 C(=O)(C(C)(C)CCCF)N1CC(COC)(NC(C2CC2c2cccc(F)c2)=O)C1 C(=O)(C(C)CS(C)=O)N(CCNC(c1n[nH]c(C)c1Br)=O)C(C)C c1(C(=O)NC(C2OCCN(C(CCNC(COC)=O)=O)C2)C)cc(O)cc(Cl)c1 N1(C(C(C)=CC)=O)C2COCC1CN(C(c1ncc(Br)cc1F)=O)C2 N1(C(C(C)(C2CCC2)NC(=O)C(C2CC2)C2CC2)=O)CCCC2(CC(O)C2)C1 N1(C(C)=O)CCCC(F)(C(=O)NC(c2csnn2)C)C1 C1(CNC(c2c(C)nc(O)s2)=O)CC2CCC(C1)N2C(C1CCN(C)C1=O)=O C1(C(=O)NC2(CCOC)CCCC2)CC2CN(C(C3CCC(=O)NC3)=O)CC2C1 Cn1nc(C(=O)NC(C2CCCCC2)C(=O)NCC2CCC(=O)NC2)cc1C#N c1(C(N2CCC(CCCCNC(CCS(C)=O)=O)CC2)=O)cnc2cccnn12 c1(C(C2CCN(C(C3CCCC4C3C4(F)F)=O)C2)=O)c(F)cc([N+](=O)[O-])cc1F C1(C(=O)NCC(C)CNC(=O)Cn2ncc(C#N)c2N)CC2CSCC(C1)C2 c1(C(N(C2CCCCC2NC(=O)C(C)(C)C(N)=O)C)=O)ccc(Cl)c(O)c1 Cn1cnc2c(C(N3CC(CNC(=O)CC(C)(C)O)C3)=O)n[nH]c2c1=O Cc1cc(C(=O)NC2CN(C(C3CCCC3(C)C)=O)CC2O)cc(C)c1Cl C(C)(CN=c1ccnc(C)[nH]1)(CC(C)C)NC(c1cccc(S(CC)=O)c1)=O C(C1COC(C)(C)O1)=CC(=O)NCCC1CCN(C(C(CC#C)O)=O)C1 CC1CC(=O)NC1C(=O)NCCCCn1cc(CN(c2ccccc2)C)nn1 N(C1CCCc2ccoc21)C(C(CC(C)(C)NC(CCC1(C)N=N1)=O)F)=O C1(NC(c2cn(CCO)nn2)=O)CCC(C(=O)NC2CC2(c2ccccc2)C)CC1 N1(C(CCCOC)=O)CCC(F)(F)C(CNC(C2CC2c2ccc(C)s2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(C3C(=C)C3)=O)C2)c(F)cc(Cl)cc1F CC1CN(C(c2cc(C3CC3)on2)=O)CCC1C(=O)NCC1=CCCN(C)C1 C1(C(=O)NCCN(C)CC)C(C2CC2)CCN1C(=O)Cc1cncn1C CCC(CO)C(=O)N1CC(O)(CCNC(=O)C(n2nnnc2C(C)(C)C)C)C1 c1(OC)ccccc1CC(=O)N(CCNC(=O)C=CCO)CCc1ccccc1 N1(C(C2CCN(CC(C)C)C2)=O)CCC(F)C(NC(=O)CCSCC(N)=O)C1 CCCCCCCN(CC(C)(C)SCC)C(c1ccc(OCCC(C)C)cc1)=O c1(OC)cc(Cl)c(Cl)cc1CNc1c[nH]nc1C(=O)NCc1nnn2ccccc12 c1(OC)cc(C(=O)NCCN2CCCOCC2)ccn1 CC1N=C(NC(=O)C2CCc3ccccc32)c2c1cccc2.N1CCc2nocc2C1 c1(C(N2CC(C(N3C(C(=O)OC)COCC3)=O)NCC2)=O)cc(Br)cc(C)c1F CCN=c1ccc(C(=O)NCCC2CN(C(c3csc(CC)n3)=O)C2)c[nH]1 CS(=O)(=O)c1ccc(C(N2CC(CNC(C34C(=O)C5CC3C4C5)=O)C2)=O)cc1 c1(C(=O)NCC2CN(C(C(CCCC#C)C)=O)CC2O)ccc2c(c1)NC(=O)C2 N1(C(C(C)NC(=O)CC(F)(F)F)=O)CCC(NC(=O)C(F)=CC2CC2)CC1C Cc1[nH]cc(C(N2CCC(F)C(NC(c3c[nH]ccc3=N)=O)C2)=O)c(=O)c1Cl C(N=c1[nH]c(=N)[nH]c(=NCc2cc(-c3ccccc3)on2)[nH]1)C1CCN(CC)C1 N1(C(CNC(=O)OC)=O)CCC2(COC(CNC(c3cn(C)nc3O)=O)C2)C1 C1(C#N)(C(N2CCC(c3c(CNC(COC)=O)c[nH]n3)C2)=O)CCCOC1 CC1CCOC1CC(=O)NC1CCCC1CN(C)C(C1CCOC1C)=O C12(C(NOCCCCC)=O)CC(CO1)N(C(=O)Cc1ccsn1)C2 C1(C(C(=O)N(CCNC(C(C(C)C)SC)=O)CCOC)O)CCS(=O)(=O)CC1 C1(C2CCOCC2)(C(N2CC3C(Nc4cc(COC)nc(C)n4)C3C2)=O)CC1 CC1(C)C(C(=O)NC2CCC2)CC1CO.C(=O)(C(CCO)NC(=O)OC(C)(C)C)N CCCCC(CC)CC(=O)NCC1(F)CCN(C(c2c(C(C)C)n[nH]c2C)=O)C1 N1(C(C2N(C(COC)=O)C(C3CC3)CC2)=O)CCC2(CC1)CSC2 c1(CCC)cc(C(=O)N(C(C)CNC(=O)C(C)(F)c2ccccc2)CC)ccn1 N1(C(C2(SC)CN(C(C3Cc4nccn4C3)=O)C2)=O)CCOCC(O)C1 C=CCC(CC(C)C)C(=O)NC1CC12CCN(C(=O)C(F)CC)CC2 N1(C(C)=O)CCC(C(N2CCCC(CN(C(=O)C=CC3CCCO3)C)C2)=O)CC1 C(=O)(CCCCC(F)(F)F)NCC(CNC(c1c(Cl)cnc(CC)n1)=O)C C=C(C)CC(C(=O)N1CC2CC1CC2O)NC(c1ccsc1Cl)=O C1(NC(COCCC#C)=O)C(C)CN(C(c2cnc3ncccn23)=O)CC1C C(=O)(CC(C(F)(F)F)NC(C1(C)CCN1C(c1ccccc1)=O)=O)OC c1(C(CC(=O)N(C2CCN(C(C=CC)=O)C2)CC)C)ccc2c(c1)OCCO2 N1(C(c2c(CC)cns2)=O)CCCC(NC(=O)CCN(C)CC)C1C C(=O)(C(C)(C(C)C)SC)NCC(CNC(c1cc(C(=O)OC)oc1C)=O)(C)OC N1(C(CS(C)(=O)=O)=O)CCN(C(c2cccc3oncc23)=O)C2COCC12 O=C1CCC(C(=O)NCCc2n[nH]cc2C(=O)NCC2(O)CCOC2)N1 C1(NC(C2CCS(=O)(=O)CC2)=O)CC2(C1)CC(CNC(C1CC3CCC1O3)=O)C2 C12(C(=O)NC(C)C(C)NC(=O)CCCCCF)CC3CC1C2C3O c1(C(=O)NC(C(N2CCCC(OC)C2)=O)(C)C2CCC2)cc(=O)n(C)cn1 CC(C)C(CCN(C(=O)C(C)(O)c1ccccn1)C)NC(C1(C)CC(C)(C)C1)=O C1(C(N2C(CC(C)C)CC2)=O)CCC(C)(C)N(C(=O)CCc2conc2C)C1 CCC(CN(C)C)C(=O)N(CC(=O)NC(c1ccn(C)n1)C)C S(=O)(=O)(c1cccc2c(C)c(C)[nH]c12)N1C(CC)CC(C)CC1 c1(C(=O)N(CCO)C2CC2)cc(C(=O)NC(c2nc[nH]n2)C2CC2)[nH]n1 c1(N2CC=CC(NC(c3c(OC)cc(Cl)cc3)=O)C2)nc(C)nc(C)c1F C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(C(C)NC(c2ccc(Cl)c(F)c2F)=O)C1 c1(OC)cc(NCc2ccc(-c3ccc(F)cc3)o2)c(Br)cn1 C1(NC(=O)CCCn2cccc2)CCC(O)C1O.C12CCC1C(=O)NOC2 Cc1ccnnc1CNC(=O)C(C1CCSC1)OC.c1(CNCCO)ccccc1Cl C1(C(=O)NCCCOCCCC)OCCC1NC(C1CCC1C)=O C12CCC(O1)C(=O)C2=O.C1(C(=O)NCCN)CC2CC2C1.C1(CC2CC2)CCC1 CC1CC(NC(=O)C=Cc2cc[nH]n2)CCN1C(c1cc(Cl)ccc1F)=O C1(C(N2CC(CNC(c3csc(C4CCCO4)n3)=O)C2)=O)CCCC1C1CC1 CC1Oc2c(C(=O)N=c3ccn(-c4ncccc4F)[nH]3)cccc2C1C N1(C(CCC(C)(C)C)=O)CC(NC(C2CCCCC2F)=O)C2(CCC2)C1 C(=O)(C(C)(C)CCC#N)N1CCCC(CNC(CNC(c2c(C)occ2)=O)=O)C1 C(=O)(CCCCCNC(C1CCCO1)=O)N(CC)CC c1(C(N2CC3(CN(C(c4c(C(C)C)[nH]cc4)=O)C3)C2)=O)nnc2n1CCCCC2 N1(C(C=CC=CC)=O)CC2CCC(C1)N(C(c1cn(C)nc1Cl)=O)C2 N1(C(COC2(C)CCC2)=O)CC2(CC2)CC1CNC(c1cnns1)=O c1(CNC(=O)CN(C)C(C2CC(C#N)C2)=O)cnc2ccccn12.Cc1nscn1 C12(CNC(c3cn(CCNC(c4c[nH]c(=O)cn4)=O)nn3)=O)CCCCC1C2 N1(C(C2OCCC(NC(C(CC)(C)CC)=O)C2)=O)CCC2(CCN(C)C2)C1 C(=O)(C1CCCn2c(C)cnc21)NC1CC(F)(CNC(C2(CC)CCCC2)=O)C1 Cc1nn(CCS(=O)(=O)N2CCCC2Cc2cn(-c3ccccc3Br)nn2)c(=O)o1 N1(C(=O)CCCOc2ccccc2)CCOC(c2ccccc2Br)C1 c1(C(=O)OCC)coc(CNCC(C2CCCO2)O)n1 C1(CNC(c2c(CC)n[nH]c2)=O)(CO)CCN(C(=O)CCC2CCC(=O)O2)CC1 N1(C(CC(C)(C)O)=O)CCc2c(NC(c3cccs3)=O)cccc2C1 C12(NC(=O)C=Cc3cccc(O)c3)CCCC1CN(C(C1CCOCC1)=O)C2 c12ccc(c3ccccc13)C(=O)NC1CCCN2C1.C1C(=O)N1.C1(NOC)CC1.O C1(CNC(CCCCC)=O)CCN(C(C2COC(=O)N2C)=O)CC1C N1(Cc2c(F)ccc(C)c2)CCC2CN(C(c3c(O)cccc3Br)=O)CC2C1 CN1CC(NC(c2ccc(CNC(C3CC(N(C)C)C3)=O)o2)=O)CC1(C)C N1(C(c2ccc(C)s2)=O)CCOCC1CCNC(C1CCN1C)=O C1(C(=O)NCC2N(C(=O)CC(C)O)CCC(CC)C2)CCc2nc(C)cn2C1 c1(C(=O)NCC2C(C)(C)CCN(C(=O)CC#N)C2)ccc2c(O)nnc(O)c2c1 N#Cc1c[nH]ccc1=NC1CCN(C(c2ccc(F)c(F)c2F)=O)CC1 O=C(C#CC1CC1)NCCNC(=O)CC1(CCc2cc(C)no2)CC1(F)F C1(C(=O)NOC(CC2CC2)C(=O)NCC=CC(=O)NC)CCCC2(CC2)C1.CO C(S(=O)(=O)c1cccc2occ(Br)c12)N1C(=O)C(c2ccc(Cl)c(Cl)c2)CC1=O C(=O)(C(=O)N=c1[nH]n(C(C)(C)C)cc1C)N1CCC(N(CC)CC)CC1 N1(C(c2sc3c(c2)CN(C(C(C)=O)=O)CC3)=O)CCC2(CCC3(CC2)OCCO3)C1 CC1CC(c2nnnn2C2COC2)(NCc2ccc(Br)s2)CO1 c1(C(=O)N(CCNC(c2cc[nH]c2C2CC2)=O)C2CC2)cc(F)cnc1O N1(C(C(C)C2CCCO2)=O)CCC12CN(C(=O)C(C)NC(=O)Nc1cccs1)C2 C12COCCN(C1)C2.C1(CNC(=O)Cc2cc(CO)[nH]n2)CCCCC12CC2 C12(CNC(C3C(C=C)C3)=O)COC(CNC(c3cccnc3NC)=O)(C1)C2 N1(C(C2N(C(N)=O)CC(O)C2)=O)CCCC2(C1)CN(C(=O)C1CC1)CCO2 c1(CC(N2CC3C(C(=O)Nc4c(C)cccc4Br)C3C2)=O)cc2ccccc2o1 C#CC1(O)CC(C(=O)NCCC2CCCN2C(=O)Cc2sc(SCC)nc2C)C1 CC1(C)C(NC(=O)CCn2cccnc2=O)CC1CNC(c1ccc(CO)o1)=O c12ccc(cc1)CCN2.c1(CNC(=O)Cc2ccsc2)ncncc1F C1(CC)CN(C(C2C3CCCCC23)=O)CC1C(=O)NCc1cnco1 C1(C(=O)Nc2cccnc2)CC2OCCC2N(C(=O)CSc2ncc[nH]2)C1 CCC(CC1CCCCC1)C(=O)N(CCCNC(c1c(C)nsc1N)=O)C C1(CNC(c2c(CC)non2)=O)CC(F)CN1C(=O)C(C)CC1CCCCC1 CC(C)(C(=O)NCc1c[nH]nc1C(=O)NCCC1CCCC2CC12)C(F)F C1(C(=O)NCC23OCC(NC(C4(F)CC4)=O)(C2)C3)CCCN(Cc2ccccc2)C1 C1(CNC(c2c(C)cco2)=O)CN(C(=O)C(O)CC(F)F)C2(CCC2)C1 Cc1cccc(F)c1C(=O)NC(C1(O)CCN(C(c2coc(C(F)F)c2)=O)C1)C C1(C2(O)CCOC2)(C(=O)OCC(c2ncc(Br)cc2F)=O)CC1 c1(CC)cc(C(N2CCN(CCNC(=O)CC3CC34CC4)CC2)=O)ncn1 c1(C(N2CC(c3ccco3)C2)=O)ccc(C(F)(F)F)cn1 N1(C(CCC)=O)CC2COCC(C1)N2Cc1[nH]cnc1-c1cncc(SC)c1 c1(C(N(CCOCCNC(CSCCC)=O)C)=O)cc(C(C)=O)cn1C C1(NC(C(Cc2ccoc2)NC(C2CCC(C)(C)C2)=O)=O)CC2CC3C(C2)C13 N1(C(C2OCCN(C)C2)=O)C2CCC1CC(O)(CNC(=O)Cc1ccsn1)C2 N1(C(c2nc(C)oc2)=O)CCSCC1C(=O)Nc1ccc(-c2ccccc2)nc1 N1(C(c2nccc(C)c2)=O)CCCC(C(=O)NCCc2cc(C)n(C)n2)CC1 C(=O)(CC(C)C(C)(C)CC)NCCC1CN(C(C=CCCC=C(C)C)=O)C1 Cc1csc(C(=O)NCCC2CCC(NC(=O)Cc3sccc3C)C2)c1Cl N1(C(C(COC)OC)=O)CC(NC(c2nocc2C2CC2)=O)C(C)(C)C1 Cc1cccc2c1CN(C(=O)COC1CCN(C(C3(C)CCC(=O)NC3)=O)C1)C2 c1(C(=O)NCC(CC)NC(c2ccnc(C)c2)=O)cn2cc(C)ccc2n1 c1(C(=O)NC(N2CC(Cc3ncc(C(F)F)o3)CC2=O)C)ccc(Cl)cc1 c1(N2CCN(C(C=Cc3ncc(C)[nH]3)=O)CC2)cccc(C#Cc2ccccn2)c1 n1(CCOCC)nnnc1C(c1cc(OC)ns1)NC1CC(CC(N)=O)C1 c1(C(=O)NCCOC2CN(C(C(C)SC)=O)C2)nc2cc(F)ccc2s1 c1(C(N2CC(C)(NC(C(C)OC)=O)C2)=O)ncnc2c1c(Br)cn2C1CC1 Cn1ncc([N+](=O)[O-])c1C(=O)NCC1CCCCN1C(c1cc(Cl)nc(=N)[nH]1)=O c1(-n2c(C(O)CCS(C)(=O)=O)nc(-c3ccc(SC)nc3)n2)ccc(F)c(CO)c1 C1(NC(C2C(C)(C)COCC2)=O)CCN(C(=O)COCCN(C)C)CCC1CO N1(C(C2CN(C)C2)=O)CC(F)CC1C(=O)NCC1(CO)CC1(C)C C1(CC(=O)NCC2CCSC2)C2CCCC2N1C(=O)CC1COCC1O N1(C(=O)CN2CCCCC2)CC2(CCN(CC3CC4CCC3C4)CC2)C1 C1(CNC(C2(C)CC(C)C2)=O)(CO)CCCN(C(C2CCCO2)=O)C1 CC1CCC(NC(c2csc(CO)n2)=O)CN1C(C1NC(=O)OC1C)=O c1(C(=O)NCCNC(c2cc(C(F)(F)F)on2)=O)cccc(Cl)c1O N1(C(c2ncn(C(C)C)n2)=O)CC2(CCCC2)C1C(=O)NC1CCCSCC1 n1(CC)nc(C)cc1C(=O)NC1CCCCC1C(=O)NC1CC(F)C1 C=C1CCC(CNC(=O)CCN(CCOC)C(c2cnn(C(C)C)n2)=O)CC1 c1(C(=O)NCC(CNC(c2c(CC)con2)=O)F)ccc(C(C)C#N)cc1 N#Cc1cncc(CNC(=O)CCC2CCCN2C(C2CCC(O)C2)=O)c1 c1(C(N2C(C(C)NC(C34CC5CC3C4C5)=O)CCC2)=O)ccc2c(c1)COCO2 C1(CCNC(c2cc(C)[nH]n2)=O)CCN(C(C2C=CC=CC=C2)=O)CC1 C1(C(N(C)CC2(O)CCN(C(C3CC=CCC3)=O)CC2)=O)CC2COCC(C1)C2 N1(CCNC(=O)CC2CCN2C(C2CCC3(CCC3)C2)=O)CCc2sccc2C1 C1(C(=O)NCC=C)CCCCC1NC(=O)C=C(C)c1ccco1 c1(OC)cc(Cl)c(C(C)NC(=O)NCCN2CCC(C)C2)cc1OC N1(C(CCSCC)=O)CC2CN(C(c3cc4sccc4cn3)=O)CC2C1 N1(C(C(c2ccoc2)SC)=O)CC2CCCC(C1)N2C(=O)C(C)C1CCCC1 Cc1ccc(C#N)cc1C(=O)NC1CCCC1NC(=O)C(C(C)C)NC=O N1(S(=O)(=O)c2ccncc2)CCC2CN(c3ncnn4cc(Br)cc34)CC2C1 c1(CCC)ccc(CC(=O)NC(C)CNC(c2ccc(-c3cc[nH]n3)s2)=O)cc1 C1(C(=O)NC2C(C)CN(C(=O)C(C)O)C2)CNC(=O)CC1(C)C C1(NC(=O)CCC2CCOC2)CCN(C(C2CC3C=CC2C3)=O)CCC1CO c1(OC)ccc(C(=O)NC2CCCC(NC(=O)CN3CCC3C)CC2)cc1SC N1(C(C(C)NC(CC)(C)C)=O)CC(CNc2nccc(C)n2)CC(C)(C)C1 c1(C(=O)NCCC(=C)CNC(C2(C(=O)OC)CC=CC2)=O)ncncc1C Cc1ccc(F)cc1C(F)(F)C(=O)NC(CNC(c1c(Cl)cncc1Cl)=O)CO C(=O)(C(C)(C)C(=O)Nc1ccccc1CO)N1C(C(C)NC(=O)C2CC2)CCC1 N1(C(C(C)c2ccco2)=O)CCCC(F)(CNC(c2cc(O)ncn2)=O)C1 CC(CC(=O)N1CCC2(CC(NC(C34CCC(CC3)O4)=O)C2)C1)CC(C)(C)C c1(C(=O)NC2CC3N(C(c4c(CC)cno4)=O)C(CC3)C2)c(F)cccc1[N+](=O)[O-] C1(C(=O)NCC(C(C)C)(C)NC(=O)CC2CC2)CC12CCOc1ccc(F)cc12 N1(C(C2C(OC)C2)=O)CC(NC(=O)Cc2cncc(C)n2)CC12CCCCCC2 CCS(=O)CC(=O)NC1CN(C(=O)C=Cc2nc(C)cs2)CC1C c1(C(N2C(C)CCC(CNC(c3ccc(O)cc3)=O)C2)=O)cccc(N=[N+]=[N-])c1 C(=O)(C(F)C(C)C(F)(F)F)NCCC(C)(C)NC(c1ccnc(OC)c1F)=O c1(NC(C)=O)ccc(C(N2CC3CCC3(CNC(c3cnn[nH]3)=O)C2)=O)cc1F CCC(C)(C#N)C(=O)NC(C)(C)CC(=O)NCC1CC(=O)N(CC)C1 C1(C)(CNC(=NCC(C)C)NCC(C)(O)CC2CCCCC2)CS(=O)(=O)CCO1 C12(C(=O)NC(CCNC(CN(C(=O)OC)C)=O)C(C)C)CCC(C1)C2(C)C N1(C(C(C)(F)F)=O)CCC2(CCCC2NC(=O)CC2CC=CCC2)CC1 CC(CCNC(=O)Cc1cnccc1Cl)CCNC(=O)COc1ccc(F)cn1 c1(CC(=O)NC(CN(C(C2CC2(F)F)=O)CC)C)nnn(C(C)(C)C)n1 CC1CN(c2nn[nH]n2)CCN1C(c1coc(Br)n1)=O CC(C)CC(C)C(C(=O)NCCOCC1CC1)N1CCSCC1.OC(=O)C c1(C(N(CC(=O)N(CC(C)CN(C)C)C)CC)=O)ccccc1 c1(CC)nonc1C(=O)NC1CCC(CNC(=O)C(CC)Oc2ccccc2)C1 N1(C(C(COC)CC(C)C)=O)CC2CC(C1)CN(C(=O)CCc1ccc(C)s1)C2 c1(C(=O)NC(C2CN(C(C(CC)OCC)=O)C2)C)cccc[n+]1[O-] C1(c2n(CCC)nnn2)(Nc2cc(OC)c(OC)cc2Br)CCC2CCCC2C1 Cc1nc2cncc(C(=O)NCCCCNC(=O)C(C)OCC3CCCO3)c2[nH]1 c1(CC(=O)NCC(N2CCOC(CNC(C3CCCC3)=O)C2)=O)ccccc1Br C1(CNC(c2c(C#C)c[nH]n2)=O)CN(C)CCN1C(=O)C(F)OC c1(C(=O)NCC(CNC(CC(COC)(C)C)=O)O)nc2c(s1)CCCC2 Cc1nn(C)c(C)c1C(C)C(=O)NCC1CN(C(=O)CCn2cncn2)CCO1 CC(C)CC(O)C(=O)N1CCN(C(=O)NC2CCCCC2)C(c2ccncc2)C1 N1(C(C(C)NS(CC)(=O)=O)=O)CC2CC(C1)C2N=c1cc(C)c(C#N)c(C)[nH]1 c1(CN2CCCC2)ccnc(Cl)c1F.C12CCN(CC1)CC1(F)CCN(C1)C2=O CC(CC(=O)NC(C)CC(=O)NCC1CC1(C)C)C1CCC1 C12(C(=O)NC(C(=O)OC)C(C)C)CCC(CN(C(C3CNC(=O)N3)=O)C1)C2 N1(C(C2(C=C)CC2)=O)CC(NC(c2cn(C)nc2-c2ccsc2)=O)C(O)C1 N1(C(c2ccc(SCC)cc2)=O)CC(CNC(c2[nH]cnc2CC)=O)C2(CC2)C1 c1(C(=O)NC2C(NC(c3n(C)ncc3C#N)=O)CC2)sc2cccnc2c1Cl c1(OC2CCN(c3n(CC4ON=C(CC)C4)nnn3)C2)c(Cl)cccc1Cl N1(C(C(C(C)C)CN(C)C)=O)CCC2CCCC12C(=O)NC1C(O)C2CCOC12 Cc1c(C(=O)NCC2CC2CNC(C2(CCC(C)(C)C)CC2(F)F)=O)cnn1C c1(CC(=O)NCC(CC=C)NC(=O)CCC(F)(F)F)cc2ccccc2cc1O N1(C(c2cnnc(O)c2)=O)CCCC(N(CC2CCOCC2)CC2CCCO2)C1 C(=O)(CC(C(F)F)N(C)CC1NC2CC1CC2C(=O)OC)OCC Cc1cn2c(n1)CCC(C(=O)NCCCCNC(=O)Cc1c(C)ncnc1C)C2 C1(CNC(C(C(C)O)NC(C)=O)=O)(CO)CCCN(C(C2CCOC2)=O)C1 N1(C(CC2C(=O)NC(=O)N2)=O)C2CCC1CC(NC(C1CCOC(=O)CC1)=O)C2 c1(C(=O)NCC2CN(C(=O)COC(F)F)CCO2)ccc(Br)c(Cl)c1F C(C(CC1CC1)C(=O)NCC1(O)CCC1)NC(CC=C)=O N1(C(C2CC2CNC(C23CCC(C2)C3)=O)=O)CC2(CCCCC2)C1 N1(C(CC(C)SC)=O)CCC2(CC1)CC2NC(c1sccc1OC(F)F)=O CC(CCCC(=O)N1CCCCC1c1n[nH]c(CO)n1)N(C)C c1(C(C)N(CC(=C)CC)C(C)C2CC2)cc(C)ccc1OC C1(COC)CN(C(C2CC(C(C)C)=NO2)=O)CCN1C(=O)Cc1cc(CO)on1 C(=O)(CCCC(C)(C)C#N)N(C1CN(C(C2(F)CCC2)=O)CC12CC2)C C1(C(=O)NC(CC)CNC(c2cc(Cl)c[nH]2)=O)CCC2(CC1)CNC(=O)C2 c1(C(=O)NCC(CC(C)C)NC(C(CC)(C)O)=O)cnc(OC)cc1C(F)F Cc1ccc(C(=O)OCC2COc3ccccc3O2)cc1S(C)(=O)=O C1(NC(C(=Cc2ccco2)C)=O)CCCC(CNC(C2C(C)C2C)=O)C1 C1(NC(c2c(C)c[nH]n2)=O)CC2CC1CN(C(C1CCC(C)CC1)=O)C2 CC1CCN(C(c2csc([N+](=O)[O-])c2)=O)CC1CNC(=O)Cn1cc(N)cn1 C1(C(C)NC(C(C)NC=O)=O)CCCN1C(=O)C1CC1 C(C(C)CC(C)C)NC(C1(CC)CN(C(C2C(C)(CC)C2)=O)C1)=O C1(CS(=O)(=O)NC2CCOC2)CCC12CCCCC2 N1(C(C(CC)(C)O)=O)CCC(C)(C)C(CNc2cc(C)ccc2OC(C)C(=O)O)C1 c1(CC(N2CCCC(N(C(c3c(C)nsc3)=O)C)C2)=O)cccc(F)c1F N1(C(c2c(-n3cccn3)cccc2F)=O)C2CCC1c1ccccc12 C(C(C)(C)C#CC(=O)N1CCC(C)(O)C1)NC(C=CC(=O)N(C)C)=O C(=O)(C(=O)C(C)CC)NCCN1C(=O)C=CC1.CC c1(CS(N2CC(n3cc(CCC(C)C)nn3)C2)(=O)=O)cccc(C(=O)O)c1 c1(C(C(=O)NCC2N(C(C(F)OC)=O)CC2)C)cccc(F)c1 CCC1=NOC(C(=O)N(C(CNC(C2(C3CCC3)CC2)=O)C2CC2)C)C1 n1(CCC)ccc(CNC(c2ccncn2)c2nnnn2C(C)C)c1 Cc1cc2c[nH]nc2cc1C(N1CCCN(C(C2(C)CC=CCO2)=O)CC1C)=O N1(C(C2C(C)OC(C)(C)O2)=O)CC23CCCC2(C1)CN(C(=O)CSCC(F)F)C3 CC(C)CC(F)C(=O)N(C1CN(C(=O)C=CC(=O)NC2CC2)CCC1O)C C1(CN(C(C2OCC(C)(C)C2)=O)CCO)COc2ccccc2O1 c1(C(=O)NC(CC)CNC(C2CC(CF)C2)=O)cc2scc(C)c2[nH]1 N1(C(CC(=O)OC)=O)CCC(CNc2cc(OC)cc(Cl)c2)C(F)(F)C1 N1(Cc2c(OCC)c(F)cc(F)c2)CCC2OCCNC2C1 C1(NC(c2c(C)coc2)=O)CCN(C(c2ccc(CN=[N+]=[N-])cc2)=O)C(C)C1 c1(CC)nc2sc(C)cn2c1C(N1CCCC1CCNC(=O)C(O)P(C)(C)=O)=O c1(C(N(CCCN(C(C=C(CC)C)=O)C)C)=O)ccc(OCCN(C)C)nc1 C=CC(F)(F)C(=O)N(CC(CO)(CO)NC(C1CCC1(C)C)=O)C C1(C(N(C(CC)CNC(=O)CC2CCCCCC2)C)=O)CC(=O)C12CCCC2 N1(C(C=CC(C)C)=O)CCC(O)C(NC(c2ccn(CCO)c(=O)c2)=O)C1 N1(C(C2(CC)CC2)=O)CC2CCC1CC2NC(C1(C2CCC2)CCC1)=O C1(C(N(C)CC2CC(O)C(O)C2)=O)N(C(=O)Cc2cc[nH]c2)CCC1(C)C C(c1cncc(O)c1)=CC(=O)NCCN(C(CN1CCC(C)C1)=O)C(C)C CC(CC(N)=O)C(=O)NC1CC(C)CN(C(=O)Cc2csc(Cl)c2)C1 c1(C(=O)NC(CCNC(CCc2ncc(C)[nH]2)=O)C(C)C)cn2ccnc2s1 N1(C(C=C(CCC)CCC)=O)CC=C(C(C)(C)C(=O)NC(C)C(=O)OCC)C1 c1(Cc2cn(C(C)CNC(C3CCC(C)(C)OC3)=O)nn2)ncn2c1CCC2 O(NC(=O)CC1CC(NC(c2cc[nH]n2)=O)C1)C(C=C)C C(=O)(C1=C(C#N)CCC1)NCC1C(NC(c2c(C)n(C)nn2)=O)C1 CCCCCCC(C)CC(=O)NCC1CCCN1C(=O)CC1CCOCC1(C)C CC(C)(C(=O)NCC1(CCNC(C2CCC(C(F)F)NC2=O)=O)CC1)C(C)(C)C CC1CCc2[nH]c(=NCCC(C)(C)C)nc(N3CCOC(c4ccco4)C3)c2C1 C(=O)(CCCCCC(C)(C)C)NCCC1CCCN(C(C(CC)OC)=O)C1 CC(C)C(C)(C)C(=O)N1CCC(CNC(=O)C(c2ccc(Cl)cc2)C)C1 C(=O)(CC(C)(C(F)F)N(C)C)NC(COC)C(C)O c1(C(=O)NC2C(NC(c3c(C)n[nH]c3)=O)CCOC2)cc(F)c(Cl)cc1Cl C1(CC(=O)N(CCC(=O)NC2CCOC2CC)CC)CCC(=O)NC1 N1(C(CCc2ccc(C)s2)=O)CC(CNC(=O)C(F)C2CCC2)CC12CCC2 N1(C(c2cc(OC(C)C)ncc2)=O)CCC2(C1)CN(C(=O)C(F)(F)C(F)(F)F)C2 Cc1nn(CCC(=O)NC2CN(C(=O)Cc3ccco3)CC2F)c(C)c1C N1(C(C(C)n2ccnn2)=O)CC(C2CC2)(C(=O)NCCCS(C)=O)C1 c1(C(=O)NC(C(=O)N(CCC#C)CCO)CCN(C)C)cccc2[nH]ncc12 c1(C(N(C(CC)CC(=O)NC(c2cccnc2)CC)C)=O)cc([N+](=O)[O-])c[nH]1 C(C)(C)(CCCC(=O)NC1CC(N(C)C)C1)NC(C(N1CC(C)C1)C)=O C#CCCCCCC(=O)OCC(=O)NC(c1cccc(C(F)(F)F)c1F)C c1(CC)n[nH]c2ccc(C(=O)OC)cc12.N12CCC(CC1)NC2=O.C1(=O)CN1 C1(C(N2C(C(N3CCC(C)C3)=O)CCC2)=O)CC2OC1C1CC21 C#CCCCCCCC(=O)N1CCC(F)(C(=O)N(C)Cc2cnco2)C1 C(c1cc(Br)cs1)=CC(=O)NC(C(C)NC(C1CC1(C)C)=O)CO CC1OC2CCC1(C(=O)NCC1CC(C(=O)NCCCN(C)C)=NO1)C2 C1(N(C(c2c(C)nsc2C)=O)C)CCCN(C(=O)Cc2cccnc2)CC1 C1(CNC(c2cn(C)nc2C(F)(F)F)=O)CCN(C(=O)CCCC2CC2)C12CC2 c1(C(N2CC(O)CC(NC(=O)COC(F)(F)F)C2)=O)ccc2c(c1)CCOC2 N1(C(c2c(N)non2)=O)CCCC(NC(=O)CN2CCCCCC2)C(F)C1 N1(C(CC2C(CN)C2)=O)CCC(C)(NC(=O)Cn2cncn2)C1 N1(C(C2CC(C#N)C2)=O)CC2CCCN(C(c3ncc[nH]c3=O)=O)C2C1 C1(C)(C(=O)NC2CC(CCC(=O)N(CC(C)(C)O)CC(N)=O)C2)CCCS1 CCC(CC(=O)NCC(c1ccccc1)NC(c1nc(O)c(C)s1)=O)CC(C)C c1(OC)cc(F)ccc1C(C1CC1)NC(=O)Nc1c[nH]nc1-c1ccccn1 N1(C(c2cnc(C)nc2)=O)C2CCC1CC(NC(C1CC3(CC3)C1)=O)C2 c1(-n2c(CC(CC)C)nc(C3CC34CC4)n2)ccc(Br)c(C)c1 c1(NC(=O)NCC(C)CNC(=O)CN(C)CC2CC2)cnc(OC(F)F)cn1 C(c1cccnc1)=CCNC(C(CNC(c1cc(OC)no1)=O)O)=O CCN=c1[nH]cc(C(=O)N(C)CCOCCNC(C2(C3CC3)CC2)=O)s1 CCCCC(CNC(c1cnsn1)=O)NC(c1cnns1)=O N1(C(CCSC)=O)CCN(C)C(C(N2CCC2C(C)O)=O)C1.C(C(C)C)O N1(C(CSCCC)=O)CCC(C)C1CNC(=O)C(CO)c1ccccc1 C=CCC(C(=O)NC(c1cccc(Cl)c1)CNC(C1(CC)COC1)=O)NC(C)=O c1(N2CCC(N(C)CC)C2)nc(=NC(CCOC)C(C)C)[nH]c2ccsc12 C(=O)(C1=CCCN(C(=O)Cc2ccc(F)cn2)C1)N(CCCC(F)(F)F)C c1(CC(C)(C)N(CCC2CCC(N)C2)Cc2ccccc2Cl)ccc(F)cc1 C1(C(=O)NCC(C)NC(c2ccc(C(N)=O)[nH]2)=O)CN(C)CC1C(F)(F)F N1(C(C=Cc2c(C)cccc2)=O)CC2CN(C(C3C4CCC(F)(F)C34)=O)CC2C1 Cc1nc2ncccc2cc1C(=O)NCCN(C)C(C1C2COCC12)=O c1(C(=O)NCC2C3CN(C(c4cnc(SC)s4)=O)C2C3)cc(F)c(C)cc1Cl CC(CCCOCCO)NC(CCCC1CC1)c1nnnn1C(C)(C)C N1(C(C=CCC)=O)CCC(NC(=O)Cc2cc(OC)ccc2F)C(O)C1 N1(C(c2cc(CC)[nH]n2)=O)CCC(CNC(C2CN(C(C)C)C2)=O)C1(C)C N1(C(Cc2cc(C)no2)=O)CC(C)(C)CC1CNC(=O)C=CBr C#CCC(C(=O)N1CC(C(N2CC(OC(C)C)C2)=O)C(C(C)C)C1)C1CC1 CCCCCCCCC(C)CC(=O)NC1(CCO)CN(C(=O)CCC(C)CC)C1 C1(CC#C)(C(=O)NCCOCCCNC(C2(CF)CCC2)=O)CCC1 C(C)(C(=O)OC(c1cccc(Oc2ccccc2)c1)C(F)F)(C(=O)O)OC C=CCC(C(=O)NC(CO)CCCCNC(c1cnc2n1CCOC2)=O)C(C)C c1(OC)ccnc(C(C)(C)CNC(c2cc(O)n(C)n2)C2CCCC2)c1 c1(CN(CC(C)NC(=O)C(=O)NC2CCSC2C)C)cccnc1 c1(CNC(=O)Cc2ccsn2)nc(CNC(=O)CN2CCCCC2=O)cc(O)n1 N1(CC(C)OC2CC(NC(=O)Nc3c[nH][nH]c3=N)C2)C(=O)CCC1=O C1(C(N2CC(NC(C3C4(CC(C)(C)C4)C3)=O)C2)=O)CS(=O)(=O)CC12CC2 C(=O)(C#CC1CCCO1)NCC1(O)CCN(C(c2cnc(COC)s2)=O)C1 C(=O)(CC(O)CN(C)C)NCC(CNC(c1c(C2C(C)C2)occ1)=O)(C)C CP(C)(=O)CC(=O)NC1COCCC1NC(c1ccnn1C1CC1)=O N1(C(CC2C(C)C2)=O)CCC(NC(=O)CCCN(C)C)C12CCC2 C(=O)(CCC(F)F)N1CCC(n2cc(C(=O)NC3(CCF)CCC3)nn2)C1 Cc1ccc(F)c(NC(=O)C(=O)NC(C)C(c2ccco2)c2ccco2)c1 N1(C(c2csc(Cl)c2)=O)CCC(NC(C23CC(CO2)C3)=O)C12CCC2 C1(NC(c2cscn2)=O)CN(C(c2cc(Cl)cnc2O)=O)CC12CCC2 C12(CNC(=O)Cc3cncc(F)c3)CCC(CC1)N(C(=O)Cc1cscn1)C2 n1(CC(=O)NC2CC(C(C)NC(=O)CSC3CCCO3)C2)cnc(C#N)n1 N1(C(c2cc(OC)cc(C)c2)=O)CCC(NC(c2cc(C)oc2C)=O)C(C)(C)C1 c1(-n2cc(CCCSCC)nn2)cccc(C(=O)NC2CCS2(=O)=O)c1 C1(N(C(c2cc(C3CC3)ccn2)=O)CC)CCCN(C(=O)CCC2OCCO2)C1 c1(OC(CC)C)ccc(C(=O)NCC2CC(NC3CCOCC3)C(O)C2)cc1 c1(C(N2C(C)(CNC(=O)CCCC3CCC3)CCC2)=O)ccc2c(c1)CCCS2 c1(C(=O)NC(C2OCCN(C(C(C)=C(C)C)=O)C2)C)cc(C)cc(C)c1C Cc1cc(C(=O)NCCCN(C(c2ccc(C(C)C)cn2)=O)C(C)C)ncc1F O=C(C1COc2ccccc21)NCC1CN(C(C2CN(C3CCC3)C2)=O)CCO1 c1(C(=O)NC(CN(C(=O)CC2CC(F)C2)CC)C)cccc(-n2cccc2)c1 n1(C(C(=O)NCC(COC)C)(C)C)cc(CC(=O)OC)cn1 N1(C(c2c(CC)ncs2)=O)CC(C2CC2)(C(=O)NCC(C)C(C)CC)C1 c1(C(=O)NC23C(CN(C(c4c(C)cnnc4)=O)C2)CC3)ccc2[nH]nc(O)c2c1 C1(NC(CCOC(CC(C)C)C)=O)CCN(C(c2cc(Cl)ccn2)=O)C1C Cc1[nH]nc(C(N2CCC2CNC(=O)CC23CCCC2C3)=O)c1[N+](=O)[O-] c1(C(CC)NC(=O)NC(c2cn[nH]c2)C)cn(C)nn1 Cc1ccc2ncccc2c1NC(C1(F)CN(Cc2cc(I)c(O)c(I)c2)C1)=O C12(NC(C=C(C)Cl)=O)CCCCC1CN(C(c1cc3cccn3c(O)n1)=O)C2 C1(NC(c2cnc(COC)s2)=O)CN(C(=O)C(C)(F)F)CC2(CCC2)C1 C(=O)(CCS(C)(=O)=O)N1CCC(C(=O)NC(CC=C)CC)(CC)C1 CCCN=C(NCC1CCC(F)(F)C1)N1CCC(c2cnccc2C)C1 C1(NC(c2n(C)nc(CC)c2Cl)=O)C2CCC1CN(C(c1cnoc1C)=O)C2 N1(C(c2cc(CC)on2)=O)CCCC2CCN(C(C3CC3c3cccs3)=O)CC12 C1(CC(=O)NC(CC)CNC(=O)CCc2ccccc2C)CN2CCN1CC2 Cc1cccc(-n2cc(-c3cc(Cl)sc3Cl)nn2)c1 C1(C(=O)NCC2(OCC)CC2)CCCCCC1NC(c1c(Cl)cnn1C)=O c1(C(N(c2ncc(Br)cc2I)C2C(C)(C)C(O)C2)=O)cc(Br)cc2cc[nH]c12 N1(C(C(C)C#N)=O)CCCCC1CNC(C1CC(OC(F)(F)F)C1)=O N1(C(c2c(CC)noc2)=O)CCCCC1C(C)NC(c1nocc1C1CC1)=O N1(C(CC=CC)=O)CCC(NC(c2nnn(-c3ccccc3)c2C)=O)CC1 c1(C(N(C(C)=O)CCc2nccs2)C)c(C)nn(CCC(=O)N(C)C)c1C N1(C2CC(C(=O)NCC(c3ccccc3)N(C(COC)=O)C)C2)CCC(C)CC1 c1(SCC(=O)NCC2C(NC(C(C)OC)=O)CCC2)ccsc1[N+](=O)[O-] c1(C(=O)NCc2cc(OC)c(OCCOC)cc2)ccc2cnnn2c1 c1(OC)ccc(C)c(C(=O)N(CCNC(=O)CCc2cnccn2)CC2CC2)n1 c1(C(N2CC3CC(C2)N(C(c2cscc2C(F)F)=O)C3)=O)ccc2n[nH]cc2n1 N1(C(c2ccn(CC(F)F)n2)=O)CC(N=c2[nH]c3ncc(Cl)cc3s2)C1 C1(NC(=O)CC2CC=CC2)CN(C(=O)C2=NOCC2)CCC12CCOCC2 C(=O)(C(F)(F)C(O)C(C)C)NCC(CC)NC(=O)Cc1cc(O)nnc1O C1(NC(=O)CSC(F)F)CCC2CCN(C(c3c[nH]cc3Br)=O)C1C2 C1(C)(CNC(C2(CC=C)CCCC2)=O)CCN(C(c2c[nH]nc2C)=O)C1 C(=O)(C(O)CCN(C)C)NC(C(C)NC(C1CCCC1C)=O)C c1(C(=O)NCC(CNC(c2cc(CCC)on2)=O)O)cccc2c1CCOC2 C(C(=O)N(C)C(=O)NCC=CCN)SCC=C c1(OC)ccc(CC(N2CCC2CNC(=O)CC(C)c2ccncc2)=O)cc1O C1(CNC(c2ccc(C(C)=O)o2)=O)C(C)CCN1C(c1ccc(CO)cc1)=O c1(C(=O)NC2CN(C(c3cncc(N)n3)=O)CC2CO)cccc2c1CCCC2 c1(C(N(C2CC(NC(=O)C#CC3CCCC3)C2)C)=O)n[nH]c2c1CCCC2 c1(CC(=O)NC2(CCNC(c3c(C)noc3C(F)F)=O)CC2)ccc2c(c1)CC2 Cc1nc2cc(NC(C3(C)CCN3C(C3CCCN(C)C3)=O)=O)ccc2o1 N1(C(CC(C)F)=O)CCCC(C2CN(C(c3conc3C(C)(C)C)=O)C2)C1 c1(C(C(N2CC(OC)(CNC(C3(F)CC3C)=O)C2)=O)C)ccccc1C CCCC(CNC(c1cnncc1OC)=O)C(=O)N1CC=C(CO)CC1 CC#CCC(C(=O)N1CC=C(C)CC1)NC(=O)Cc1ccc(C#N)cc1 CC(C)(C(=O)N1CCC(C(N2CCSCC2C2CC2)=O)O1)N1CCOC1=O.C(C1CC1)N n1(CC)nc(C(=O)NC2CC(F)(CNC(C3(C)CC3)=O)C2)cc1O n1(CC)nc(C)c(C(=O)NCC2(NC(=O)C(C)C#N)CC2)c1C N1(C(c2cnc(-c3c(C)cncc3)s2)=O)CCCS(=O)(=O)CC1C(=O)OC(C)(C)C C12(C(N)=O)CCCC1(C(=O)NC1CCC(CNC(=O)Cn3cnnc3O)CC1)C2 C=C(C)CC(C(=O)NOCC=CC)NC(=O)CCC1CCC1 c1(C(=O)NC2(CNC(C3(COCC)CC3)=O)CC2(C)C)sc(C(C)C)nc1C c1(C(N2C3C(NC(C(C)N4CCC4)=O)CC(C3)C2)=O)n[nH]c2ccc(Cl)cc12 CC(C)(C(=O)NC(CC(=O)NC1CCCC1)C(F)F)C(N)=O C1(C)(CNC(C=CCCC)=O)CC(OC)CN1C(=O)CNC(=O)C(C)(C)C c1(C(=O)NCCC(C)CCNC(c2cn(C3CC3)cn2)=O)cc(F)c(N)cc1F c1(C(=O)NCCC(CNC(C(C(CC)O)C)=O)(C)C)c[nH]c2nccc-2c1 Cc1ccc2c(c1)C(C(=O)NC1CCOCC1NC(c1cncn(C)c1=O)=O)C2 c1(OC)ccc(CCC(=O)Nc2ccccc2SC(C)(C)C)c(Br)c1 N1(C(c2sc(C)c(O)n2)=O)CC2(C1)C(NC(=O)CSc1nncs1)CCS2(=O)=O c1(OC)ccc(CNC(=O)C(=O)NCc2ncccc2C)cc1OC(F)F N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)(CNC(=O)C(C2CC2)OC)CC1 CC(C)CC(C(=O)NC1C2CN(C(C3CCCN3C(C)C)=O)CC12)N(C)C c1(CNC(CCSC)=O)cccc(CNC(C2(c3ccccn3)CCC2)=O)c1 c1(NC(C2CCCC2NC(=O)Nc2ccc(C)cc2)=O)cccc(F)c1I N1(C(C(CC)(C)CNC(c2cn(C)c(=O)cn2)=O)=O)CCC(C)C(F)(F)C1 c1(NC(c2cccc(NCc3ccc(F)cc3)c2)=O)cc(Br)cnc1O N1(C(CN(C(C)C)CC)=O)CC(C(=O)N(C2CC2)Cc2cccnc2)(C(N)=O)C1 C1(C(N(C)CC2CCCN2C(=O)CCCC(C)(C)C)=O)CC2(CCOCC2)CO1 c1(C(N2CC(C)C(NC(c3cccc(CS(C)=O)c3)=O)C2)=O)cccc(O)c1F CCC(CC)C(C)N=c1cc(Cl)nc(CN2CCCC2)[nH]1 Cc1cc(S(=O)(=O)NCC(C)C)n(CC2CCOCC2)n1 c1(CC(=O)N(C)CCNC(C2(c3cccs3)CC2)=O)ccc([N+](=O)[O-])cc1F CC(C(=O)NC(c1ccccc1)C(=O)N(C)CC1CCCN1C1CC1)C(F)(F)F N1(CC)N=C(C(=O)NCC2CC2NC(C2(C)CCC(C)(C)CC2)=O)CCC1=O C(=O)(CCCCCCNC(c1cn[nH]c1)=O)N1C(COCC#C)CCCC1 C1(CN(C(C2CCCO2)CO)C)CCN(C(=O)OC(C)(C)C)C12CCC2 c1(C(=O)NC2C(NC(c3cc(CC)c(CC)o3)=O)COC2)cc(C)c(F)c(C)c1 C(=O)(CC(O)CC(C)(C)C)N1CCCC(N(C)C(C2CCCCS2)=O)C1 Cc1[nH]c2ccc(O)cc2c1C(N1CCN(C(C2CC23CC3)=O)C(C(C)C)C1)=O c1(C(=O)NC(C(C(C)C)Sc2ccccc2)C)cc2c(s1)CCC2=O c1(C(=O)NC2CC(C(=O)NCC3CN(C)C(=O)C3)C2(C)C)c[nH]c2ccncc12 Cc1nc2ccc(C(=O)NCC3CC(NC(=O)CC(F)F)C3(C)C)cc2nc1C CC(C)CC(O)C(=O)N(C)CC1CN(C(=O)CC(C)(C)O)CC12CC2 N1(C(c2[nH]cc(C)c2)=O)CCC2CN(C(c3cc(O)cc(Cl)c3Cl)=O)CCC12 C1(NC(C2(CC)CCC2)=O)(CF)CCN(C(=O)C(C)COC(C)=O)C1 C1(C)(C(=O)NCC(C)CNC(=O)C(C)n2ccnc2)CC1(Cl)Cl C1(C(N(C)CC2N(C(C(C)SC(F)(F)F)=O)CCCC2)=O)CC2C=CC1CCC2 c1(C(COC(C(N2C(=O)CCC2=O)CC)=O)=O)ccc(N(C)C)cc1 c1(C(N(CC(CNC(COCCCOC)=O)O)C)=O)ccc(-n2ccnc2)cc1 C1(N(C(Cc2c(C)nn(C)c2)=O)C)CCN(C(C2(C#N)CC2)=O)CC12CC2 O=C(C1=CCCSC1)NC1CC2CC(NC(C3C=CCS3)=O)C2C1 c1(C(N)=O)ccsc1NC(C1CCN(C(=O)C(c2cccnc2)O)C1)=O C1(NC(C(C)Cn2cccn2)=O)CN(C(c2cnc(S)[nH]2)=O)CC1(C)C Cc1cccnc1C(=O)NC(C)(CNC(=O)CS(=O)(=O)NC1CC1)C(C)C c1(OC)cc(C(N2CCC(NC(=O)CCc3nc[nH]n3)C2)=O)c(N)c(Br)c1 N1(C(CC(=C)C)=O)CCC2(CC1)CC(CNC(=O)CSc1cnn(C)c1)C2 N1(C(=O)CCC(F)F)CC23CCCCC2(C1)CN(C(=O)CCC1CCCO1)C3 O=C(CC(F)(F)Cl)NCC(CO)NC(C1CN(C2CCCCC2)C1)=O.C(C(F)(F)F)S CC(=O)CCCCC(=O)N1CCCC1CNC(=O)CCOC1CCCCC1 c1(C(=O)NC2CCN(C(c3c(C)cc[nH]3)=O)C2(C)C)ccc2c(n1)CCC2 C(=O)(C1=C(Cl)CCOC1)N1CC(C)C(C)(CNC(c2c(F)cccc2F)=O)C1 c1(CC(N2CC(N(C(C(CC)OC)=O)C)C2)=O)cccc(F)c1OC C(=O)(C(CC)CC(F)F)NC1(CC=C)CCN(C(=O)Cn2ncc(O)nc2=O)C1 C=CCCC(C)(C)C(=O)NC1(CNC(C2CCOCC2)=O)CC1.C12CCN1C2=O c1(C(=O)NC2CCN(C(C(C)(CO)OC)=O)C2)oc2c(C)ccc(C)c2c1C C#CC(CNC(=O)C(CC(=C)C)NC(=O)CN1CCOCC1)CC(C)(C)C N(C1CCc2ccc(Br)cc21)C(C1CCN(C(c2c(C)[nH]cc2)=O)CC1)=O CC(N=c1[nH]c(N2CC(F)(F)C(F)(F)C2)nc2c1CCC2)c1ccc(Cl)c(Cl)c1 CC1(C)CCN(C(c2ccsc2Br)=O)CC1NC(=O)C1=CCS(=O)(=O)C1 N1(C(CSCCCC)=O)CC(n2cc(CNC(=O)COCCOC(C)=O)nn2)C(C)C1 O=c1c2cc(Br)ccc2ncn1CCN1CC(O)CCC1c1ccccc1CO C1(NC(C(C(C)NC(=O)CCN2CCCC2=O)C)=O)CCC(C#N)CC1 C1(NC(c2c(C)cco2)=O)CN(C(=O)C(C)CSC(F)(F)F)CC1O C(=O)(CC(C(F)F)NC(C1(C)CC2C=CC1C2)=O)NCc1cn(CC=C)nn1 c1(C(N(C)CC2C3CN(C(C(CC)(C)F)=O)CC32)=O)cnc2ccccc2n1 N1(C(c2nc(C(C)C)sc2)=O)CC(NC(C2CCCC2)=O)CC2(CCOCC2)C1 N1(C(C(C)OCC)=O)CCN(CC2CN(C(=O)C(c3cccc(C)c3)C)C2)CC1 N1(C(CCC(=O)OC)=O)CC2CCC1CN2C(=O)Cc1cc(C)sc1Cl C=CC1(C(=O)NCCOCC(C)C)CCN(C(=O)Cn2nc(C)oc2=O)C1 C1(NC(c2ccoc2)=O)CC2CCC1CC2NC(C1Cc2nnsc2S1)=O N1(C(c2sc3cccc(N(C)C)c3c2)=O)CC2COCCC2(NC(=O)C(N)=O)C1 Cc1c(F)ccc(C(=O)NCC2CCCC2C(N(C)CP(C)(C)=O)=O)c1C c1(CNC(C=C(CNC(c2nncc(OC)c2)=O)C)=O)ccc(C)c(F)c1 c1(C(N2CC(SC)C(NC(=O)Cn3ccnc3C)C2)=O)c[nH]c2cccc(C)c12 S(=O)(=O)(c1cc(Br)ccc1Br)N1CC(CC)N(c2ncnc3c(Br)csc23)CC1 C12(NC(C(COCC)NC(c3cc(C)c(Cl)s3)=O)=O)CCCC1C2(F)F C1(NC(=O)Cc2csc(C3CCCCC3)n2)CCCN(C(C2CC23CC3)=O)C1 c1(CNC2(c3nnnn3C)CC(C3C(=O)NC(=O)N3)C2)c(Cl)cc(Br)cc1Cl C1(C(=O)NCc2n(C)nnc2)CN(C(=O)COc2ccccc2)CC(C)(C)C1 N1(Cc2cc(C)c(F)nc2)CC(C(N2CC3CC2CN3C)=O)CC(F)(F)C1 c1(NC(CC2CC(N(C)C)C2)=O)cnn(CCOC(C)(C)C)c1 CCC(C(=O)NNc1cc(C)c(Cl)cn1)NC(C1CCCN1C(=O)OC)=O C=CCC(C(=O)NCC(C)(Cn1cccn1)NC(=O)CN(C1CC1)CC)C(C)C C1(C(C)C(=O)N2CC(OCC(=O)N(CCO)CCC3CCCC3)C2)CCC(=O)N1 c1(-c2cc(C(=O)OC)c(OC)nc2)cc(S(=O)(=O)NCC(F)F)ccc1OC C1(C(=O)NC(CC)CNC(c2cc(F)ccc2O)=O)CC2CCC1C21CC1 C1(CNC(C2C(C#N)CC2)=O)CC12CCN(C(c1csc(Cl)n1)=O)CC2 C1(NC(C=Cc2cc(C)no2)=O)C2CC1CN(C(=O)CCn1ccnc1)C2 CC1(C)COCC(C(=O)NCCN(c2ccccc2)C(c2c[nH]ccc2=O)=O)O1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(O)(CNC(=O)CN2CCNC(=O)C2)C1 O=C(C1CCCc2nn[nH]c21)NC1CCN(C(c2ccoc2Cl)=O)CC(O)C1 O=C1NCC(C(=O)NCC2(O)CC(C(=O)NCC3NCCCS3)C2)O1 C1(Cn2cc(CSCC)nn2)CCN(C(=O)C(N2CCSCC2)C)CC1 CC1CCN(C(C23CCCN(CCC2)C3)=O)CCN1C(C1CC(=O)N1)=O C(=O)(C(C(C)CC)NC(=O)C1CC1)NC(CC1CCN(C(C=CC)=O)CC1)C c1(-c2c(OC)ccnc2)nc2c(s1)CC(C(=O)Nc1ncc(Cl)cc1Br)CC2 CCC(CC(=O)NC(C)CC1CN(C(=O)C(c2ccccc2)N(C)C)C1)C(C)C c1(C(=O)NC2CC(NC(c3nc(COC)sc3)=O)C2)cc(=O)c(C)c[nH]1 N1(CC)CC2CN(C(C3CC(C(=O)O)C34CCC4)=O)CC2C1 C(=O)(C1=CC2CCCCC12)N(CC(C)NC(CCC=C(C)C)=O)C CC1CC(CC(=O)NCC2CC2)CN1C(c1ccns1)=O.C1C(=O)N1 c1(C(N2CCC2c2ccc(Br)cc2)=O)cc2c(-c3ccoc3)cncc2s1 C(=O)(CN=S(C)(C)=O)N1CCCC(N(C(CCC(C)N(C)C)=O)C)C1 N1(C(C)=O)CCCC(c2cn(CC(C)O)nn2)(NC(C2CCSC2)=O)C1 C(=O)(C(F)(F)CCn1cccn1)NCC1C(NC(CCC(=O)N(C)C)=O)CC1 C1(CNC(C2CC(OCC)C2)=O)CCCCC1N=c1ncnc2[nH][nH]c(C)c1-2 C(C)(C)(CC(=O)NCC12CC1CN(C(c1cc(C)nn1C(CC)CC)=O)C2)OC C1(CC)CN(C(C2CCN2C(=O)OC)=O)CCC1N(C)C(C)=O c1(-c2n(C)ccn2)ccnc(N2CCC(CNC(c3ccc(F)cc3)=O)CC2)n1 CC(C)C(F)(CNC(=O)C=CCF)C(=O)NCC1(CO)CCN(C)C1 c1(C(C)=O)cc(C)cc(O)c1.c1(-c2cn(C(C3N(C(C)=O)CCC3)=O)nn2)c(C)cnn1C C12(CNC(c3c(C)nns3)=O)CCCCC1CN(C(=O)Cc1cccc(Cl)c1)C2 CCC(C)(COC)C(=O)NC1CC2(C1)CC(CNC(C1CC(OC)C1)=O)C2 N1(C(C2N(C(c3scc(C#N)c3)=O)CC(O)C2)=O)CCc2nocc2C1 C(=O)(C(C)CC(C)(C)C)NCc1oc(C)c(C(N2CCCCCC2CCO)=O)n1 C1(n2c(CC(n3cncn3)C)nc(C3CCCCCC3)n2)CCCS(=O)(=O)C1 C1(C(=O)NC(CNC(c2ccc(CO)o2)=O)CO)CC(F)(F)CS1 C(=O)(C1CCN(C)c2ccccc21)NC(C)CNC(C1CC2CC2C1)=O C(=O)(CC(C(F)(F)F)NC(=O)C1=C(C)CCCC1)NC(COC)(C)CO CC(C)(C)C(CNC(C1CCN(CCO)C(=O)C1)=O)C(=O)NS(=O)(=O)C(F)(F)F c1(C(=O)NC2C3(CCN(C(C(C)=O)=O)C3)C2)ccc(S(=O)(=O)C(C)C)cc1 Cn1nc(C(F)(F)F)c2cc(C(N3CCC(=O)C4CCCC34)=O)sc12 C(=O)(C(C)C1=CCCC1)NCC(N1CCN(C(c2ccc(C)nc2)=O)CC1)C n1(C2CN(C(C3(CC)CC3)=O)C2)cc(CNC(c2ccnn2C)=O)nn1 Clc1ccccc1C(c1nnnn1Cc1ccccc1)NCC1CC2CCC1C2 C1(C(=O)NCC(O)CC(=O)NC(CO)C2(O)CC2)CC2(CCO1)CC2 c1(C(=O)NCCN(C(C2CCS(=O)(=O)N2)=O)C2CC2)c(C2CC2)cccc1F Cc1nsc(C(c2nnnn2C)NCCn2ccnc2C)n1 N1(C(CN(c2cc(O)n(CC)n2)CCC)=O)CCC2CCC(O)C1C2 CCCC(O)(CCC)CC(=O)N1CCN(C(=O)CCc2ccco2)CC1CF Cc1ccc(C)c(CC(=O)NC2C=CCN(C(c3nc(C)n(C)c3C)=O)C2)c1 Cc1c(Cl)cnn1CC(=O)NCC(CNC(=O)CCc1ccsc1)CO N1(C(c2cc(C(C)(C)C)no2)=O)CCN(C(C2CC2c2cn[nH]c2)=O)CC1CF c1(CNC(C(C)OCOC)=O)ncc(C(=O)NC2(CO)CCC(C)C2)cn1 N1CC2CCC1C(O)C2O.CC1CCCC=C1C(=O)N1CCC1C12CC1CNC2=O c1(C(N(C2CCCN(C(C(CN(C)C)(C)C)=O)C2)C)=O)nc[nH]c2ncnc1-2 O(NC(=O)CC(C)C(C)(C)NC(=O)CC1(O)CCOCC1)CCOC c1(C(=O)NCC(CN(C(c2c(COC)cc[nH]2)=O)C)O)ccc(CO)cn1 C1(C(=O)NC(CCCC)CNC(=O)CN2CCN(C)CC2)CC(=O)NC1(C)C C1(C(=O)NC(CCOC)CNC(C2CC2C)=O)C(C)(C)C1(C)C N1(C(CC=CCC)=O)CC(NC(c2oc(C3CC3)nc2C)=O)CC1(C)C C1(CNC(c2cc(C)c(O)nc2)=O)CN(C(=O)Cc2ccon2)C2(CCC2)C1 N1(C(C2(C(=O)NC(C)C(C)N(C)C)CC2)=O)CCCN(C(c2ccoc2)=O)CC1 c1(C(N2CC(NC(C3C(C)(C)CC3)=O)C2)=O)cc(C(F)F)ccc1F CC(O)C(F)(F)C(=O)NC1C=CC(CNC(c2cccc(-c3nnco3)c2)=O)C1 c1(C(=O)NCC(C)(C2CC2)NC(CC2C(C)OCC2)=O)coc2c(Cl)cccc12 C1(CNC(c2c(NC(CNC(=O)OCC=C)=O)ccs2)=O)CCCC1(C)CC C1(C(=O)NC2CC(C)N(C(C3CCCOC3C)=O)C2)CC2(CCCCC2)C1 C1(CC(N2CC(CNC(=O)CCCc3ccsc3)C2)=O)CCCC2CC12 C1(CCC(=O)NCC2(F)CN(C(=O)CCOC3CCOC3)C2)CC=CCC1 C1(C(=O)NCC(C)CC2CC2)(NC(=O)CCc2nccn2C)CCC(C)(C)C1 C=CCC(C)C(=O)N1CCCCC1CN(C(=O)CC1(COC)CCC1)C Cc1c(SC2(C(N3CC(NC(=O)CN(C)C)C(C)C3)=O)CC2)oc2ccccc12 c1(N(C)C)ccc(C(=O)NCC2(C)CCN(C(C3CCOCC3)=O)C2)nn1 C1(CNC(CC(C)c2cnn(C)c2)=O)CC(NC(=O)C=CCCC(C)C)CCO1 c1(OC)cncnc1C(=O)NC(C(N)=O)C(C)c1ccccc1 c1(C(=O)NCCNC(C2C=CCC2)=O)cccc(CO)c1.C1(C(=O)N)CCCC1CF C1(NC(CSCC#C)=O)CCSC12CN(C(C1CCn3ccnc3C1)=O)C2 C12(CNC(C=CC=CC)=O)CC1CN(C(=O)C(C)Oc1ccccc1F)C2 C1(C)(C(=O)OC(C)C(=O)Nc2cc(Br)cnc2Br)CCC(F)(F)CC1 C1(C(=O)NCC2C(CNC(CC3(COC)CC3)=O)C2(F)F)C=CCCC1C C1(C(=O)NCCS(CC)(=O)=O)CCC(O)CN1C(c1cc(C(C)C)nn1C)=O c1(C(=O)NC(C)CNC(=O)CN2CC3C=CC2C3)noc2c1CC(C)(C)CC2 N1(C(C(CC)O)=O)CCc2nc(O)cc(-c3cn(-c4ccccc4)nn3)c2C1 c1(CC(=O)Nc2cccc(NC(c3c(C)ncn3O)=O)c2)ccc(F)cc1F N1(C(c2ncn(CCOC)c2)=O)CCOC(C(C)Oc2ccc(COC)o2)C1 CC1=C(C(=O)N2CC3CC(NC(c4csc(CO)n4)=O)CC3C2)CCCC1 C1(F)(C(=O)OC)COCCN(C(=O)NCc2cc(CSC(C)(C)C)cn2C)C1 C1(CNC(C(CC)=CC)=O)CCN(C(=O)CCCc2ccccc2)CC1O C1(C(=O)NCc2cc(C(=O)NCC(C)(CO)OC)on2)CCCC(=O)CC1 C#Cc1cnc(C(=O)NCC(C)CNC(c2c(OC)cccc2F)=O)c(C)c1 C#Cc1cn(C)nc1C(=O)N(C(C)CN(C)C(c1scnc1COC)=O)C C(=O)(C1CCCc2ncc(C)n21)N(CC(C)O)CCNC(C1(CC=C)CC1)=O Cc1c(C(N2CCCC2C(C)(C)C(=O)N(C)Cc2ccncn2)=O)cccc1O CC1OC2(C)CC1(C(=O)NCC1CCC(CNC(=O)Cc3ccn(C)n3)CC1)C2 c1(C(=O)NC2C(CNC(=O)CCc3ccon3)CCCC2)ccc([N+](=O)[O-])[nH]1 CC1(C(=O)NC2CN(C(c3ccc([N+](=O)[O-])o3)=O)C2)CCC2CC2C1 C1(NC(c2n(C)ccc2)=O)CC2CCC(C1)N2C(c1cocc1C(N)=O)=O c1(C(N2CCC(N(C(Cc3c(C)nc(C)s3)=O)C)C2)=O)c(F)ccc(F)c1Cl C1(NC(CCC(=O)N(C)C)=O)CC2CC1N(C(=O)Cc1cccc(Br)c1Cl)C2 Cc1cc(C)c(C(N2CC(C)(NC(C3(c4ccccc4)CC3(C)C)=O)C2)=O)n1C c1(C2N(C(c3ccsc3Br)C(=O)NC(C(=O)OC)C)CC2)ccc(F)cc1 N1(CC2ON=C(C(C)C)C2)CCN(S(C)(=O)=O)CCC1C C(C(C)(C)C#CC(=O)N1CCCOCC1C)NC(CCCCC#C)=O N1(C(c2c(C)noc2C)=O)CC2CCCCC2(NC(=O)CCCCN(C)C)C1 C1(C(N)=O)COC2(CCN(C(C3CC3c3cncc(Br)c3)=O)CC2)C1 C1(CNC)CN(C(c2cccc(C(F)(F)C(F)(F)Cl)c2)=O)CCCO1 C1(NC(=O)CCC2CCC2)CCN(C(C2CC2F)=O)C12CCC2 C1(C(N2CCN(C(C3=C(C)CCC3)=O)CC2CCO)=O)CCCC2CCCN12 Cc1ncc(C(=O)NCC2CCN2C(=O)C(O)CC2CCCCC2)cc1Cl N1(C(c2cc(CC)[nH]n2)=O)CC2CN(C(=O)CC3C=NN(C)C3=O)CC2C1 C1(C(=O)NCCCC2(NC(CCC#CC)=O)CC2)CC12CCOc1ccccc12 c1(OC)ccc(Cl)c(C(=O)NCCN(C(=O)Cc2cncn2C2CC2)C)c1 C1(NC(CCC(=O)NC)=O)CCN(C(c2ocnc2C(C)C)=O)CC1C S(=O)(=O)(c1csc(C(=O)NC(C2CCCN2C(=O)C(C)=C2CC2)C)c1)NC CC(C)C(O)CC(=O)N(C)CC1CCCN(C(C2(C)CS(=O)(=O)C2)=O)C1 N1(C(CN(CC)CC)=O)CCCN(C(=O)COC2CCOCC2)CC1C(C)C N1(C(CSCCC)=O)CCC(NC(=O)C=Cc2cnc[nH]2)CC1c1ccccc1 c1(C(N2CCCC(NC(C(CSC)O)=O)(CO)C2)=O)c(N)ccc(C)c1F c1(OC)c(C(=O)NCC(C)(C(C)C)NC(c2cn(C)cn2)=O)oc2ccccc12 Cc1coc(C(=O)NCCCCC(C)NC(=O)C(c2ccc(F)cc2)F)c1C N1(C(c2n(C)cnc2)=O)CC2CCOC2(CNC(=O)CCc2ccsc2)C1 CCCC(CNC(c1coc(COC)n1)=O)NC(=O)C(O)C1CCC1 C#CCC(C(=O)N1CC(CC(=O)NCCn2cc(Cl)cn2)(OC)C1)C1CC1 C1(CN(N2C(N)CCC2)C)CCN(C(C2(c3cccs3)CC2)=O)C1.C(=O)C1CC1 Cc1cnc(NCC2CCCC(NC(C3CC34CC4)=O)C2)nc1 C(=O)(C(F)C(C)(F)F)NCc1ccc(C(=O)NC(c2cccc(O)c2)C)cn1 CC(C)S(=O)(=O)C(C)C(=O)NCC1C(C2CC2)CCN1C(C1CCCC1C)=O CC1OCC2(CCN(Cc3cccc(F)c3N)CC2)C1NC(=O)C1=COCCO1 c1(OC)c(C(N2CC(N(C(=O)C(C)OC)C)C2)=O)cccc1[N+](=O)[O-] N1(C(C(F)OC)=O)CC(CNC(=O)Cn2nccn2)C(O)C1 C(=O)(CC(CNC=O)CC(C)C)NCCCCC(CO)NC(CC(=O)OC)=O CCCC(C)(O)CC(=O)N1CCN(C(C2(S(C)(=O)=O)CC2)=O)CC12CC2 CCCC(CCCNC(=O)Cc1ccon1)NC(=O)C(C)(C)c1ccns1 c1(OC)ccc(Cl)c(C(=O)NC(CNC(=O)Cc2nnc(C)o2)C(C)C)c1N FC1(F)CC12CC(NCc1cnc(C3CC3)o1)C2 C1(CNC(C=Cc2ccc(C)o2)=O)CC2(CC2)CN1C(C1CC2CC1C1CC21)=O c1(C(=O)NCCOCCN(C)C(C2CC2(C)C)=O)cccc(-n2cnnn2)c1 Cc1ccc(C(=O)NCC2CCCC3CC23)c(-n2cc(CC(O)C(C)C)nn2)c1 C#CCC(C(=O)NCC(C)(C)CO)NC(C1CN(CC)CCO1)=O N1(C(C(C)NC(N)=O)=O)C2CCC1CN(C(c1ccncc1Cl)=O)CC2 c1(N2CC(=C(CNC(CC)=O)F)C2)nc(Cl)nc(OC(C)CC)c1C#N C12(NC(c3[nH]c4cc(C)oc4c3)=O)CCOCC1CN(C(c1scnc1Cl)=O)C2 c1(NC(=O)NCCN2CCN(C(C(=O)OC)C)CC2)cc(F)c(Cl)cc1Cl C1(C(=O)NCC2(NC(c3cc(C#N)[nH]c3)=O)CC2)CCOC2(CCC2)C1 c1(C(=O)NCCN(C(C(CC)C2CCOCC2)=O)C)nn(C)cc1Cl N12CCOCC(C1)C2=O.C1(NC=O)CCc2ccoc2C1.Cc1ccccc1CO c1(N(C)Cc2cncc(F)c2)nnc(C2CCOC2)n1CCOC1CCSCC1 c1(C2(NC(C(C(C)(C)O)F)=O)CCCC2)nnc2ccccn12 c1(C(C(=O)NC2(CC)CN(C(C(C)OCC#C)=O)C2)O)ccccc1Cl CN1CCCC2C1CCN2C(=O)Cc1csc(-c2ccsc2)n1 Cc1ccc(N2CCC(c3ccc(C(N4CCCC4=O)=O)cc3)CC2)nc1C c1(CC(=O)NC2C3CN(C(c4ncc(NC)nc4)=O)C2C3)cnn2ccccc12 C1(C)(NC(C2N(C(CCCOCC)=O)CC2)=O)CCC(C)(C)C1 c1(NC(CCC)CCC)nc(C)cc(=NC2CC3C(C2)C3(F)F)[nH]1 c1(C(=O)NC2(C)CCN(C(CN(S(C)(=O)=O)C)=O)C2)cc2c(Cl)nccc2s1 Cc1cc(CCC(=O)NC2CCC(NC(C3CCC(C(N)=O)O3)=O)CC2)nn1C O(NC(=O)C(c1ccccc1)NC(=O)COC1CCCC1)C(C)C C1(CC=C)(C(=O)N(C2CCCC2)C)CN(C(=O)CC2CC(N(C)C)C2)C1 C=CCC(C)(C)CNC(C1COCCN1C(c1cc(C)oc1CC)=O)=O C(=O)(C1CCCn2cnnc21)NC1C(C)CN(C(=O)C(F)=CC2CC2)CC1 Cc1cccc2c(C(=O)NC3CCN(C(C4C5CNC(=O)C45)=O)C3)coc12 C(=O)(CCCC(=O)c1ccccc1)N(C)CCNC(=O)C(O)Cc1ccccc1 Cc1ccc(-c2noc(C(C)NC(=O)C(N3CCC(CNC4CC4)C3)=O)n2)cc1 Cc1cc(C2CC2)ccc1C(=O)NCCOC(c1ccccc1)=O c1(-c2ccc(CCCCCC)cc2)n[nH]c2c1CN(C(=O)C(C)(C)CN(C)C)C2 n1(CC(N2CCCC(CCNC(=O)COCCCF)C2)=O)ncc2cccnc12 N1(C(C2(C3CCCC3)CCC2)=O)CCCCC1CNC(CNC(C1C(C)C1)=O)=O n1(CCC(=O)NC(C2(C(=O)O)CC2)C)cc(C2CCCOC2)nn1 N#Cc1cc(F)c(C(=O)NCCCCNC(=O)CCOCC(F)F)c(F)c1 C1(NC(CC(CC)SC)=O)CN(C(=O)CN(C(=O)C(C)C)C)CC12CCOCC2 C12(C(=O)NCCC)COCC1CN(CCCc1ccc(Cl)cc1F)C2 c1(C(N2CC(CNC(=O)CC3CCOC3)C(O)C2)=O)ncc(Br)cc1F N1(C(c2c(Cl)cc(C)c(C)c2)=O)CCC2CCN(C(=O)C(F)C(F)(F)F)CC2C1 Cc1nc2c([nH]1)C(C(=O)NC(C)CCNC(=O)CCc1ccc(C)o1)CCC2 N1(C(C=CCC)=O)Cc2ccnn2CC(NC(=O)C(c2ccc(C)cc2)(F)F)C1 C(=O)(C1=C(Cl)CCC1)NCC1C(NC(CC=C=C)=O)CC1 C1(C(=O)NCC2CCN(C(CN(C3CCCC3)C)=O)C2)CCCOCC1 C(CCCCC(=O)NOCC(N1CCCC(C)(C)C1CO)=O)OC C(CCC(O)C(=O)NCC1CNC(=O)C1)NC(C=CCC)=O N1(C(c2occ(C)c2)=O)CC(CNC(=O)CC2OCCCO2)CC(C)C1 c1(C(C)=O)ccc2c(c1)CN(C(c1sc3ccc(C#N)cc3c1C)=O)CCO2 c1(C(=O)NC2C3C(C)N(C(C4CC=C(C)CC4)=O)C2C3)cn2cccc(C)c2n1 C1(C(=O)On2c(C3C(C(=O)OC)C3)nnn2)(CCC2CCCO2)CCCC1 CC1(C)CCC(C(=O)NCc2cc(C(=O)NC3CCCC(F)C3)cs2)C1 C1(F)(CNC(=O)Cc2cc(Cl)ccc2Cl)COCCN(C(C2CNC(=O)C2)=O)C1 C1(C(=O)OCC)CCN(C(C2CC3CC3C2)C(=O)N(CCCC2CC2)C2CC2)C1C N1(C(C2C(C(C)C)C2)=O)CC2CS(=O)(=O)CC2(NC(c2ccsc2)=O)C1 C1(CCN(C(=O)CCc2nccs2)C)CCCCN1C(c1cccc(CO)n1)=O n1(CC)nc(C2CC2)cc1C(N1CC(CN2CCCC2)C1)=O.n12cc(nn1)CS2 c1(C(=O)NC23C(CN(C(c4c(C)occ4)=O)C2)CCC3)cc2ccsc2c(O)n1 c1(C(=O)NC2CCN(C(CS(=O)(=O)NC)=O)C2)csc(S(C)(=O)=O)c1 c1(C(N)=O)cnccc1CNC(CN(C(=O)COCC1CC1)CC)=O C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCC(O)(CNC(CC(C)c2ccsc2)=O)CC1 CCCC(C(=O)NCCCCF)NC(=O)CN(C)C C(CC(=O)NCc1cccnc1C)(CC(C)C)NC(C(CC=CC)CC)=O c1(NCc2cccc(C3(S(C)(=O)=O)CC3)c2)cc2cn[nH]c2cn1 n1(CCC(=O)NCC(C)(C)CNC(=O)C(O)CF)cnc2ccccc12 CCC(C)C(O)C(=O)NC(C1CCN(C(=O)C(O)Cc2cnc[nH]2)CC1)C N1(C(C=CCC)=O)CCCC(C(=O)N(C)Cc2ncn(C)n2)C1C C(=O)(C(F)(F)C(F)F)N1CCC(N(C(C(C)OC)=O)Cc2ccncc2)CC1 c1(C(N2C(C)CC(NC(=O)CC(F)(F)F)C2)=O)ccc2c(O)nccc2n1 C1(NC(C2(CCCC)CCC2)=O)CSCC1C.C12CC1C(=O)N2 N1(C(C=CCC)=O)CCC(CC(C)NC(=O)CC(C)COC)CC1 c1(CNC(=O)Nc2cnc(Cl)nc2)noc2c1CCCC2 C1(C)(C(=O)NC2C(CNC(CCCNC(C)=O)=O)CC2)CC(C2CC2)=NO1 CC1Cc2cc(S(=O)(=O)NCc3ccc(OCC(=O)O)cc3F)ccc2O1 c1(C(N(C(C)C)CCNC(=O)C(O)C2CC2)=O)cc2sc(Cl)cc2[nH]1 C1(NC(C(CC)NC(N)=O)=O)CCC2CCN(C(c3ncccn3)=O)C1C2 c1(C(N2C(C)(C)C(NC(=O)COCCO)CC2)=O)cc(F)cc2ccncc12 c1(C(C)NC(CNCC(C2CCCC2)OC)=O)ccc(C#N)cc1 C1(C(=O)NC(CC=C)C2CC2)(C(C)C)CCN(C(=O)C(C)(Cl)Cl)C1 C(CCCCN(C(=O)CC1CCCSC1)C)NC(C=C(COC)C)=O C12(NC(COCC)=O)CCCC1CN(C(c1cc(-n3cccn3)ccn1)=O)C2 N1(C(CSCC(N)=O)=O)CCCC(NC(c2ccn(C3CCOCC3)n2)=O)C1 c1(N2CC(C)(NC)C2)ncnc(NC(=O)CSc2nc(-c3cccs3)n[nH]2)c1C Cc1ncc(C(=O)NCCC23CCC(C2)N(C(C2(CC4CC4)CC2)=O)C3)c(=N)[nH]1 C1(NC(=O)CC2CCOCC2)CCCCCN(C(C2CC(C3CC3)=NO2)=O)C1 C=CCCCCC(=O)N1CC(C)(C)CC1CNC(C1COC2COCC12)=O C1(O)(C(C)NC(C=CC=CC)=O)CN(C(C2CC2C(F)(F)F)=O)C1 C(=O)(CCCC(=O)N(C)C)NCC(C)NC(C1(c2ccncc2F)CCC1)=O C1(CC(=O)N(CC(=O)N(CCO)CC2CCC2)C(C)C)CCOC1C C12(NC(CC(CCCC)O)=O)CC3CCC(C1C2)N3C(c1ccc(=N)[nH]c1)=O c1(C(C)(C)C(=O)NCCc2cn(CC3CC3C(F)(F)F)nn2)ccc(Cl)cc1F C1(CNC(c2c(C(C)NC(c3ccc(C(N)=O)[nH]3)=O)noc2)=O)CCCC1(C)C c1(CC(COCOCC2CSCCN2Cc2ccccc2)C=O)ccc(F)cc1F.CO CC1(C(N2CCCC(CCNC(c3ncc[nH]c3=O)=O)C2)=O)CC2CCC(C1)S2 CC1Oc2ccccc2OC1C(=O)N(C)CCN(C)C(c1cnc(O)c(Cl)c1)=O CCCCC(C)(C)NC(=O)C(F)CC1CN(C(=O)Cc2ccccc2F)C1 c1(C(=O)NC2C3CN(C(C4=CC(C)(CC)C4)=O)C2C3)cc(F)c2nc(C)cn2c1 c1(C(N2C(C(C)NC(=O)CCc3ccc(F)cc3)CCC2)=O)ccc(O)c(F)c1F c1(N2CC(C)(CNC(CC(=C)C)=O)OCC2)ncnc2cccc(Br)c12 c1(C(=O)NCC2N(C(CCC(C)SC)=O)CCCC2)ncnc(O)c1Br CC(C)CCC(O)C(=O)N1CCC(C(N)=O)CC1.C1(=O)C(F)C2(CCC2)N1 C(=O)(CS(=O)CCC(F)(F)F)NCCCN(CCCNC(C1(SC)CCC1)=O)C N1(C(c2scc(COC)c2)=O)CC(NC(C2C3CCCC23)=O)CCC1C C(=O)(CCCC(F)(F)F)NC(C)CCCCNC(=O)CN(C1CCSC1)C N1(C(C(C(CC)O)C)=O)CCOC2(CCCN(C(c3cc(O)nn3C)=O)C2)C1 C(=O)(CCC(C)(C)C#N)NC(CC(=C)C)C(=O)NCCCc1cccnc1 O=C(CCCC(F)(F)F)NCC1CC1CNC(C1CCC(O)C1)=O C(=O)(C1=NNC(=O)C1)NC(C1CN(C(c2cc(Cl)cc(Br)c2)=O)CCO1)C C(=O)(CCCC(=O)NC1CC1NC(c1scc(C)c1OC)=O)NCCC C1(C(=O)NC(C)CNC(C(=O)NCC2CC2)=O)CC12CCC(C)(C)CC2 C=C1CCN(C(=O)OC(C)(C)C)C(C(=O)NCC(C)OC(C2CCN(C)CC2)=O)C1 N1(C(c2n(C)cnc2)=O)CCN(C(C2CC2CF)=O)CC1c1cc(F)ccc1F c1(C(=O)NCCN(C(=O)CCCOC(C)(C)C)CCC)cnn(CC)c1C c1(C(N2CCC(NC(c3c(C)onc3O)=O)CC2C)=O)ccc2c(c1)CCN2C N1(C(C(c2cn(C)nn2)NC(CCn2ccc(C)n2)=O)=O)CCC2CN(C)CC12 C1(OC(c2c(C)n(C(C)C(C)(C)O)nc2)=O)CC2(C1)CC(c1ccccc1)C2 c1(CCC(=O)NCC(CC)NC(c2cc(C)c[nH]2)=O)ccc(Cl)cc1 C1(Cl)(C(=O)NC2CC(NC(c3c(C(C)C)[nH]cc3)=O)CC2O)CC12CCOCC2 c12cccc(c1)NC2c1nnnn1CC1CCCO1.c1(SC)cncnc1 N1(C(c2occ(C)c2)=O)C2CCC1C(CO)N(C(c1cccc(N)c1)=O)C2 c1(CC(=O)NCC2CCN(C(c3cccs3)=O)CC2O)cc(F)cc(Br)c1 CCCC(CCCNC(=O)C(C1CCC1)OC)NC(c1cc(CC)[nH]n1)=O C(=O)(C1=C(CC)OCCS1)N1CCC(F)(CNC(c2c(F)ccc(CC)c2)=O)C1 c1(C(C)C)nnc(C=CC(N2CC3CC3(NC(=O)CC3CCC(O)C3)C2)=O)o1 C12(NC(=O)CCCc3ncco3)CCCCCC1N(C(=O)Cc1cnns1)CC2 CN1CC=C(CC(=O)N2CC3CCCC3(NC(=O)CC(=O)NC3CC3)C2)CC1 c1(C(=O)NCC(C)CNC(c2cnc(CC3CC3)s2)=O)ccc(Br)c(F)c1 N1(C(C2=CCCC2C)=O)C2COCC1CN(C(=O)CN1CCC(C(N)=O)CC1)C2 c1(OC)c(C(=O)NCc2cc(C(=O)NCCC3CC(O)C3)n[nH]2)cnn1C Cc1cc2cc(C(N3CC(C)N(C(c4n[nH]cc4C)=O)CC3C)=O)c(Cl)cc2[nH]1 c1(C(=O)NCC2CC(O)CN2C(N)=O)c[nH]cc(F)c1=O.C12CCN1C(=O)C2 c1(C(=O)NC2CN(C(COC(CC)C)=O)CC2C)ccc2c(c1)CCC2 CS(=O)(=O)C=CC(=O)NCC(C1CCN(C(c2cccnc2O)=O)CC1)(C)C C1(C2(O)CN(C(=O)CCC3CCCC3)C2)(CNC(=O)CN2CCCS2(=O)=O)CC1 C1(CNC(N(CCCCO)CC)=O)CCN(C)C1 c1(NC2CC(CNC(C(C)NC(C)=O)=O)C2)ncc(C#C)cn1.C1C(=O)N1 c1(C(=O)Nc2cc(C(F)F)ccc2[N+](=O)[O-])ccc2c(c1)CNC2=O C(CC(=O)N=S(C)(=O)c1cccnc1Cl)OCc1c(C)cc(C(F)(F)F)cc1 c1(C(N2CC(CN(C(C(C=C)(C)O)=O)CC)OCC2)=O)ccc(C)cc1C1CC1 N1(C(c2c(CC)nccn2)=O)CCN(C(c2sc(=N)[nH]c2C)=O)CC1CC O=C1CN(C(c2ccc(F)cc2)=O)C(C(N2CCCC2CF)=O)CN1 CC(C)C(C)(CNC(C1(C)CC=CCC1)=O)NC(=O)COC1(C)CCOCC1 Cc1cc(C(=O)NC(C)(CNC(c2c(C)noc2C2CC2)=O)CO)ncc1F C12(CCNC(=O)CC3(NC(C4COCOC4)=O)CC3)CCCC1C2 C12(C(N3CCC(CN(C(CS(CC)=O)=O)C)CC3)=O)OCCCC1C2(F)F Nc1ccc(C(=O)NCC2(CNC(c3cc4scnc4[nH]3)=O)CC2)cc1F C1(C2CC2)(C(=O)NC(C2N(C(C3N(CCC(C)C)CCC3)=O)CCC2)C)CCC1 c1(OC)ccc(C=CC(=O)NC2(C)CN(C(c3cccc(CSC)c3)=O)C2)cc1 N1(C(c2cn(CCNC(C=C(COC)C)=O)nn2)=O)CC(C)C12CCOCC2 c1(CCC(=O)NCCCN(C(=O)CC(C)(C)CC=C)CC)c[nH]c2cc(Cl)ccc12 C(CCCCC(=O)NC1CC2(C1)CC(NC(=O)CNC(N)=O)C2)NC(C)=O CCCC(C)CC(=O)NCCN1CCCN(C(C2(CO)CCCCO2)=O)CC1 C1(C(N(CC(C2CC2)OC)C)=O)CC2(CC2)CN1C(c1cnc(C)[nH]1)=O C1(NC(CCC(=O)NCC)=O)CN(C(C2CCOC2)=O)CC1(C)C C(CC1=CCN(CC=CCl)CC1)N(C(=O)C(F)(F)F)C(CSS(C)(=O)=O)=O CN1C(=O)CCC1C(N1CCC(F)(C(N2CCC(CF)(CO)C2)=O)C1)=O C(=O)(CCC1=NNC(=O)CC1)NC1CC(C)(CNC(Cn2ncn(C)c2=O)=O)C1 c1(C(=O)NCC2(F)CCN(C(CNC(C(CC)C)=O)=O)C2)sc2nccn2c1C CC1CN(C(=O)C(C)(C)C2CCC2)CC1NC(C1CCCN1c1ncccn1)=O N1(C(C2C(C)(CC)C2)=O)Cc2[nH]nc(C(=O)N(C)CC3CC3(F)F)c2C1 N1(C(CCC(=C)C)=O)CCC2(NC(=O)C3=NOC(C(C)(C)C)C3)CCCC12 N1(C(CNC(C2CC(NC(COC)=O)C2)=O)=O)CCC(O)C(C)C1 Cc1ccn(C(C)CC(=O)NCC2CCN2C(=O)CCc2cn(C)cn2)n1 c1(NC(C(c2ccccc2)SC)=O)cccc(S(N)(=O)=O)c1.N12CCCC(C1)C2 C1(NC2(c3nnnn3C3CC3)CCC=CCC2)C(C2CC2)CCN1CC1CC1 Cc1cc(=NC2CC2Nc2ccccc2)[nH]c(N2CC3CCC(C2)C3O)n1 C1(CC)CN(C(=O)C(C)(C)COC)CCN1C(=O)C(CCOC)c1ccccc1 C1(OC)C2CC3C(C2)C13C(=O)NC1CCOCC1F N1(C(C(c2c(OC)cccc2)=O)=O)Cc2nccn2CC(C)C1 c1(C(=O)NC2(CN(C(C(CC(C)C)O)=O)C)CC2)ccc2oc(O)nc2n1 CCCC(C)(CC)C(=O)NCC1(C)CC(NC(c2cn(C)nc2Cl)=O)C1 C1(C(N2CCC(C(F)F)(CNC(C(C)N3CCC3)=O)C2)=O)CCC2(CCC2)C1 c1(C(=O)NC(C2(O)CCN(C(=O)Cn3ccnn3)C2)C)ccc(N)cc1O C1(CC)CCN(C(c2ccn(C)c2)=O)C(C(=O)Nc2cccc(CO)c2C)C1 N1(C(c2c(C)onc2-c2ccccc2F)=O)CC2(CCN2C(C2CC2F)=O)C1 CN1CC(C)(C(=O)NC2CC(CNC(C3C=CCCC3)=O)C2)CC1=O n1(CC(N2C(CNC(C(CCC)C#N)=O)CCC2)=O)ccc2ccc(F)cc12 C1(O)(CNC(=O)CCC2CCC2)CCCN(C(=O)CC2CCCCC23CC3)C1 N12CC(C(F)(F)C1)C2=O.c1(CC)cnccc1C(=O)NC1CC1.C12(CC1)C(=O)N2 CCC(CC)(CO)C(=O)NC1CN(C(=O)CCc2cccc(F)c2F)CC1F N1(C(C(=Cc2ccco2)C)=O)CC2(CNC(C3CC3CF)=O)CCC1CC2 CCCCC(C(=O)NCCC(N1CCOCC(O)C1)=O)NC(N)=O c1(C(=O)NC2(C)CC(NC(C3CCn4cnnc4C3)=O)C2)ccc(S(N)(=O)=O)s1 C12(NC(c3c(CC)cccc3)=O)CCC(C1)N(C(C1CC(OC)C(OC)C1)=O)C2 c1(NC(C(C)Oc2ccc(Cl)c(Cl)c2)=O)cc2cc(Br)ccc2[nH]1 C1(C(=O)NCCCCNC(c2csnc2C2CC2)=O)CC2CC1CO2 c1(OCC)ccc(S(=O)(=O)N2CCCC2C(=O)Nc2cnn3c2CCCC3)cc1 C(=O)(N=c1[nH][nH]c2ncccc12)C1(C)CCN(C(c2cccnc2)=O)CC1 C1(CNC(c2cn(CC)nc2)=O)CN(C(c2n[nH]c(C)c2C)=O)C2CC12 C(=O)(CCCCCF)NCCC1CC(C(=O)NCC2ON=C(CC)C2)C1 c1(OC)cc(NC(=O)C(=O)NC2CCCC2(C)CSC)nc(C(F)(F)F)n1 C(=O)(C(F)(F)C(F)F)N(C)CC1(CNC(=O)CC2CCCS2(=O)=O)CC1 C(C(O)CC(=O)N1CCOC(C(=O)NC2(C)CCCCC2)C1)N(C)C c1(C(=O)NCC(CC(C)C)NC(Cc2c(C)noc2)=O)ccc2ccnn2c1 c1(C(=O)OC(c2nc(C)sc2C)=O)nc2nc(C)ccn2n1.N1(CC)CC1.CC N1(C(CCC(C)O)=O)CC2CN(C(=O)CN3CCOCC3)CC2C1 C1(OC)CCC2CN(C(C3CCCCCN3C(C34COCC3C4)=O)=O)CC12 C1(SCC(CC)Oc2ccccc2F)CCN(C(c2cc[nH]c2)=O)CC1 C1(NC(CCn2ccc(C)n2)=O)CCCCN(C(c2cnn(C)c2F)=O)C1 C(C(C)CC(=O)NCC(c1ccc(C(F)(F)F)cc1)O)OC C1(NC(CSCCN(C)C)=O)CCCN(C(=O)Cc2nn(C)cc2Br)C1 c1(N(C(c2cnc(C)n2C)C(=O)OC)C2CCC2O)ccc(C=CCO)cc1F Cc1cc(C(=O)Nc2ccc(Br)cc2I)cc2c1CCC2 c1(C(=O)NC(C)CN(C)C(C23CC(C)C2C3)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 N1(C(c2[nH]cc(C)c2C)=O)CCC(O)(CCNC(c2c(CO)noc2C)=O)CC1 c1(C(=O)NCC2(F)CN(C(Cc3cc(C)cc(F)c3)=O)C2)cc([N+](=O)[O-])cn1C N1(C(C2C(C#C)C2(C)C)=O)CCCC2(C1)CN(C(c1coc(CO)c1)=O)C2 c1(CNC(C2CCCS2)=O)cccc(CNC(C2CCCC3CC23)=O)c1 C1(CC=C)(NC(=O)CCC(C)SC)CCN(C(=O)CCCN2CCCCC2)CC1 C1(NC(C(C)NS(CCC)(=O)=O)=O)CN2CCC1CC2 N1(C(CNC(CN(C)C)=O)=O)CC(O)(CNC(=O)CC2(C)CC2)C1 C12(NCc3cccc(OC)c3)CC(CNC(c3ccc(C)o3)=O)(C1)OC2C C1(NC(c2scc(C)c2C)=O)CC2CCC(C1)N2C(=O)Cc1ccno1 N1(C(C2(CC=C)CC2)=O)CCCC(C2CCN(C(C3C=CCC3)=O)CC2)CC1 C1(NC(c2c(O)cccc2F)=O)CN(C(=O)C=CC2CCCO2)CC12CCC2 C(CC(=O)NC1CC1NC(=O)CC1CCSCC1)(C(F)(F)F)OC c1(NC(=O)Nc2cc(C(=O)OC)n(C)n2)ncc(C)cc1[N+](=O)[O-] C(N=c1[nH]c2c(c(=NCCC3CC3)[nH]1)CSC2)c1c(C)ccc(C2=CCCC2)c1 C1(O)(CCNC(c2nc(OCC)sn2)=O)CCN(C(=O)CC2CC2)C1.C(=O)(N)NC N1(CCNC(C=C(C)C(C)(C)C)=O)CCCN(C(C2CCCCN2C)=O)CC1 N1(C(c2cccc(NC(N(C)C)=O)c2)=O)CCN(C(=O)CP(C)(C)=O)C(CO)C1 c1(C(=O)OC)cccc2sc(C(=O)NCC(C)(C)NC(C3C4CCCC34)=O)cc12 c1(CC(C(=O)N(C)CC2(OC)CCOCC2)N)cc(Br)ccc1O c1(C(N2CC(N(C(C3C(C)C3)=O)C)C(O)CC2)=O)cc2c(ncn2C)s1 c1(CC(N2C(C(CNC(CCC=C)=O)(C)C)CCC2)=O)cccc2cn[nH]c12 c1(C(=O)NC2CCN(C(c3occ(C)c3)=O)C2C)ccc2nc(C)nn2c1 S(=O)(=O)(c1cnc(NCCCC2CCOCC2)c(Cl)c1)N(C)CC1CC1(C)C c1(OC)n[nH]c(C(=O)NCC2(CNC(C3(C)CCC(=O)N3)=O)CCCC2)c1Cl N1(C(C(C)Cc2cccnc2)=O)CCn2ncc(CNC(=O)C(O)C(F)F)c2C1 C=CCCC(C(=O)NC1CCSCC1)NC(=O)CNC(C1CC1C)=O C(=O)(C1=NNC(=O)C1)NC1(C(N2CCC(O)(CC(C)C)C2)=O)CCSC1 C1(CNC(C2Cc3nncn3C2)=O)CC12CCN(C(=O)Cn1nccn1)CC2 CC1(C)CN(C(=O)CC2(O)CCOCC2)CC(C)(C)C1NC(C1CC1C(N)=O)=O CCC(F)(F)C(C)(C)C(=O)NCCN(CC(C)O)C(c1ncoc1C1CC1)=O C(=O)(N=c1cc(C)n(CC(=O)OC)[nH]1)N1CCC(C)(CCC#C)CC1 c1(OCCC(=O)NC2CN(C(C(CC)COC)=O)C2)ccc(Br)c(C)c1 C1(CC)CN(C(C2C(C)(C)OC2(C)C)=O)CCN1C(C1CC1C(F)F)=O Clc1cc(Cl)ccc1-n1ncnc1-c1ccccc1.C12(CCCC1)CC(CN)NC2 C(=O)(C1CCCc2ncnn21)N1CC2(CCN(C(c3cnc(C)n3C)=O)CC2)C1 c1(CC(C)C(=O)NCC2(NC(=O)CC3CCCO3)CC2)cccc(F)c1 c1(C(=O)NC2(C)CCN(CC#N)CC2)ccc(S(C)(=O)=O)cc1.O(NC)CC C(CC(F)F)(C(=O)NOC1CCOCC1)NC(c1cccc(=O)o1)=O C1(CNC(c2c(C)cc(C(F)F)o2)=O)CCN(C(=O)CNC=O)C(C)C1 N1(C(c2c(Cl)cccc2Br)C)Cc2ccccc2C(NC(=O)OC(C)(C)C)C1 Cc1ccncc1CNc1c(I)cnn1C(C)(C)C N1(C(Cc2ccc(OC)o2)=O)CC2CCC1CN2C(C1(N(C)C)CC1)=O C(=O)(C(CCCC)NC(c1csnc1OC)=O)NCC(C#C)CC C1(F)(CNC(=O)NC(c2ccc(C)cc2)CO)CCC(C(=O)OC(C)(C)C)CC1 CCC(O)C(C)C(=O)NCC(C1CCCCN1C(c1ccoc1C1CC1)=O)(C)C C(C(C(=O)N1CC(C)C1C(=O)NCC1C2COCC12)OC)OC C1(CC)CN(C(=O)CSCC(C)=O)CCN1C(C12CCC(COC)(C1)OC2)=O N1(CC(C)C)N=C(C(=O)NC(CNC(=O)C(C(C)C)C(C)C)CO)CCC1=O N1(C(C(C=C)(F)F)=O)CC2CCN(C(c3nocc3CC)=O)CC2C1 C(C1=NOC2CN(C(c3ccsc3C#N)=O)CC12)NC(c1cc(C(C)C)no1)=O C=CCCCC(C(=O)N1CC2CC(O)CC2C1)NC(=O)C=Cc1cnccn1 C(CC(C)CC)(C(=O)NC1(C#C)CCOC1)NC(c1n(CC#C)ccc1)=O c1(C(N2CC(C)N(C(C3(C)CC3)=O)CC2)=O)nc2ccc(Br)cn2c1N c1(C(=O)NCC2CCCN2C(C2CCC(F)CC2)=O)c(O)ccc(F)c1F C1(C(CO)NC(C2(C)CCC(C)C2)=O)CCN(C(c2ccc(OC)s2)=O)CC1 C1(C(=O)NCC2CC23CCC3)CCC(NC(COCCCOC)=O)CC1 N1(C(CSc2cccc(OC)c2)=O)CCC(CO)C(NC(=O)C(C)(F)F)C1 C(c1ccc2c(c1)CCO2)=CC(=O)NC(C1CCN(C(=O)CCN2CCCC2)C1)C CC(F)(F)CC(=O)NCC12CC1CN(C(=O)CSCc1ccc(Cl)cc1)C2 c1(OCC)ccc(Cl)c(C(=O)NCCCCNC(c2ccn(C(C)(C)C)n2)=O)n1 Cc1noc(Cl)c1CC(N1CCC1CNC(=O)CCN1CCCCC1)=O C(=O)(C(C)(C)CN(C)C)NCC(CC=C)NC(C1CC(C)CCO1)=O C(=O)(C1CCCc2ccnn21)N1C(CNC(CN=S(C)(C)=O)=O)CCCCC1 Cc1cc(Br)cc(F)c1C(N1CC(C)(C(N2CCN3C(=O)CCC3C2)=O)C1)=O Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(C)(C)Cc2cnn[nH]2)cn(C)c1=O N1(C(C(C)=C(CC)C)=O)CC(C)(OCC(=O)NCC2(Cl)CC2(F)F)C1 Cc1[nH]nc2ncc(C(N3CCC4CC4(NC(c4cc(F)c[nH]4)=O)CC3)=O)cc12 C(C(=O)NCCC(O)CNC(c1csc(-c2ccccc2)c1)=O)(C(C)C)OCC n1(CC)nncc1C(=O)NCc1cc(C(=O)N(C)CC2CCSC2)co1 C1(C(N(C2CN(C(C(COC)OC)=O)C2)C)=O)Cc2ccccc2N1 Nc1c(C(=O)NCC2CC2NC(C2CC3CCC2O3)=O)cccc1Br N1(C(c2cnsc2)=O)CCCC2(CCN(CCc3cc(F)cc(Cl)c3)C2)C1 c1(C(=O)NCC(CNC(C(CC)OC)=O)O)cc(C)n(-c2cccnc2)c1C C1(C(=O)NC(C2(O)CCCCC2)C)CC(O)CN1C(=O)CCC1(C)CC1 C1(C(N2CC3C(NC(c4c(CC)nco4)=O)C3C2)=O)CCc2cnnn2C1 c1(C(=O)NC(CCCC)CNC(=O)C(C)COC)cc(C(N)=O)cc(F)c1 c1(C(C2CC2)NC(N2CC(C#CC)C2)=O)ccc(Br)c(F)c1C C1(NC(CCCC(=O)NCCC)=O)CN(C(=O)C(C)N2CC(C)C2)CC2(CC2)C1 c1(NC(C2OCCN(C(c3scc(C)c3Cl)=O)C2)=O)ncc2cc(Br)ccc2n1 CC1COC2(C1)CN(C(C1CN(C(=O)OC(C)(C)C)CCC1(C)C)=O)C2 N1(c2cccc(C)c2)CCN(C(=O)N(c2cc(C(N)=O)ccc2C)C2CC2)CC1=O CN1CC(NC(=O)C(C2CCN(C(c3cnn(C)c3)=O)C2)F)C(=O)N1 c1(-n2c(C(CCOCC)NCCc3cc(C)[nH]n3)nnn2)c(C)cccc1C C[Si](C)(C)C#Cc1ccc(NS(=O)(=O)c2cc[nH]n2)cc1 c1(C(N2CC(CC(C(=O)NCC(C)N(CC)CC)F)C2)=O)cnn(C)c1C C1(NC(c2c(CNC(C3(SC)CC(=O)C3)=O)cco2)=O)CC(=O)N(O)C1 C1(CCNC(Cc2c(C)nc[nH]2)=O)CCCN(C(=O)COC2CCCCC2C)C1 C(CN=c1[nH]cc(C(N)=O)s1)C1OCC(C)C1 N1(C(c2cc(C)[nH]n2)=O)CCN(C(c2cc(-c3ccc(C)s3)[nH]n2)=O)CC(C)C1 C1(NC(CCc2cnc(C)s2)=O)CCN(C(=O)Cc2ccon2)CC1C(C)C N1(C(c2cn(CCC)nc2)=O)CCC(C(CO)NC(c2ccc(=N)[nH]c2)=O)CC1 CCCC(CC(C)C)C(=O)NCC1(C(=O)NC2(C)CC(C)(C)C2)CC2(CC2)C1 Cc1ccc(Nc2ncc(C3CC3)cc2Br)c(C)c1 N1(C(c2n(CC)cnn2)=O)CCC2CCCN(C(c3ccc(Cl)c(C)c3)=O)C2C1 c1(C(N2CC(c3c(CNC(C4(OC)CCOC4)=O)ocn3)C2)=O)ccc(=N)[nH]c1 c1(OCC)ccc(C2(C(=O)N(CC(C)(C)CNC(=O)C(CC)SC)C)CC2)cc1 N(C1CSCc2ccccc21)c1cc(C)c(NC(=O)C(N2CCOCC2)=O)cc1 c1(C(N2CC(NC(C(C(C)C)NC(C)=O)=O)C2)=O)cn(C)c(=O)cn1 C(C)(CN=c1ccnc(C2CCCC2)[nH]1)NC(c1cc(C)nc(Cl)c1)=O c1(C(=O)NC2CN(C(Cc3c(C)nc(C)s3)=O)C3C2C3)ccc2nc(O)[nH]c2n1 N#Cc1ccnc(N2CCC(NC(=O)C=CC3CCCO3)C2)n1 CCC(CC)C(C)C(=O)NC1COCC1C(N1CCC(CO)C(C)(C)C1)=O c1(C(N2CC(CNC(C3(F)CCCC=C3F)=O)C2)=O)ccc(F)cc1Cl C1(NC(c2cccnc2S)=O)CCN(C(=O)CCCN2CCCCC2)C12CC2 C(=O)(C(C)(C)NC(=O)C(F)CC1CCOC1)N(CCCCC)CCN(C)C CC(C)C(C(=O)NC1CC(NC(=O)CCc2ccccn2)C1)N(C)C Cc1ccc(C=CC(=O)NCC2CN(C(=O)C(N3CCOCC3)C)CCO2)s1 CC(C)(O)C(C)(O)CNC(C)(CCN1CCOCC1)c1ccncc1 C1(COC)(NC(=O)CC(F)F)CCCN(C(=O)C(F)(F)CC2CC2)C1 C(=O)(CC1=CCCCC1)NCc1cccc(NC(C2(OC)CCCOC2)=O)c1 C1(NC(c2cnsn2)=O)CCC12CN(C(c1cncc(C3CC3)c1)=O)C2 C(CC(C(=O)N(C)CCc1ccccn1)NC(C1CCC1C#N)=O)OC CC(C)C1=NOC(C(=O)NCCC(O)C(=O)NC2CCCC2(C)CO)C1 CC1(C)CCCC(C(c2nnnn2C2CCOCC2)NCCCn2cc(Cl)cn2)C1 C1(NC(Cc2c(F)ccc(C)c2)=O)CN(C(c2nocc2Cl)=O)CC1S(C)(=O)=O C=CC1(CC(N2CCC(C)CC2CNC(C2(F)CCOC2)=O)=O)CCOCC1 c1(OC)ccc(C(=O)NC2(C3CCCCN3C(C3CC(=O)N(C)C3)=O)CC2)cn1 c1(C(N2CC(Nc3ccn(CCOC)n3)C(F)C2)=O)cc(Br)cc(Cl)c1F C(=O)(C(O)CC(F)(F)F)NCc1c(C(=O)NCCOCCC)nco1 c1(CC(=O)N(CC(C)NC(C2CC2C(F)F)=O)CC)ccc(-n2cnnc2)cc1 c1(CNC(CC(C(C)C)c2ccon2)=O)ccc2c(c1)C(C)(C)CN2 c1(C(C(=O)NCCCC)N(C)CC2C3CCC2(C)C3(F)F)cc(Br)cc(OC)c1F C#Cc1ccccc1CC(=O)NC1(COC)CCN(C(=O)C(C)C2CCCC2)CC1 C1(C(N2C(C)CC(NC(c3occc3Br)=O)C2)=O)CCc2c[nH]nc2C1 N1(C(CN2C(C)CC2)=O)CCN(C2CCCN(C(c3csc(CO)n3)=O)C2)CC1 Cn1cnc2cnc(NCC(C3CCCC3)NC(c3ocnc3C3CC3)=O)nc12 C=CC1CN(C(=O)CCCC(=O)N(C)C)CC1NC(=O)C(=O)N(CCC(N)=O)CC c1(C(N2CC(CNC(C(c3ccccc3)SC)=O)C(C)C2)=O)c(N)cccc1Cl N1(C(C(CC)(F)F)=O)CCC2CCC(NC(c3cc[nH]n3)=O)C1C2 c1(C(=O)NCC2(CCNC(=O)CCCC3CCC3)CC2)ccccc1Br c1(CC)cc(NC(C2CCCN2C(=O)CC(C)(C)OC)=O)cc(C)c1 C1(CNC(CC2CCC(C)CC2)=O)CCC2(CC1)CC(NC(C13CC(F)(C1)C3)=O)C2 C1(C)(C(C)C)CCN1C(=O)CC1CCC(NC(c2cc(Cn3nccn3)on2)=O)C1 C1(OC)(CO)CCC(C)(C)CC1.C1(CNC(C=C(COC)C)=O)CCC(C)CN1C=O C1(C(C)C(=O)NC2COCC2F)CCCN(C(=O)CCc2cncnc2)C1 C1(NC(C(c2cn(CC)nc2)=O)=O)CCCCC1CNC(=O)C(C)C c1(C(C)C)cc(C(=O)NC2CCOCC2NC(=O)CC2CC=CC2)c(C(C)C)o1 C1(C(=O)NCCC2CN(C(c3c(CC)cno3)=O)C2)Cc2nccn2C1 Cc1cnn(CC(=O)NOCC(N2CCCC2C(N)=O)=O)c1 Cc1c(C(N2CC(CC(=O)NC(c3cccnc3)C)CC2(C)C)=O)[nH]ccc1=O c1(N2CCC(c3ccc(C)cc3)CC2)ncnc2c1ncn2CCC1CC1CSC Cc1ccc(CCC(=O)NC2CC(C)N(C(c3ccc(=O)n(C)c3)=O)C2)cc1Cl N1(C(COC(CC)C)=O)CCCN(C(=O)C=Cc2ccsc2C(F)(F)F)C(C)C1 c1(C(=O)NCCC2(C)CCCO2)cccc(CNC2CCSC2)n1 N1(C(CC(CC)OC)=O)CC2CN(C(c3cc(C)cc(C)n3)=O)CC2C1 Clc1nc(Nc2cnn(C3CC3)c2)c2sccc2n1 O(N(CC)C(=O)NC1C(C(=O)OC(C)(C)C)C1(F)F)CC C(CCCCC(=O)N1CCC(C)(CC(=O)NC(C2CCC2)C)C1)OC C1(CC#N)CN(C(=O)Nc2cc(C(F)F)ccc2Cl)CCN1C(=O)CC#N Cc1cc(C(C)(C)C(=O)NCC(F)CNC(c2cccnc2C2CC2)=O)ccc1F c1(C(=O)NC2CCCN(C(c3cncc(C)n3)=O)C2)sc(Br)c(C)c1C CC1(C)CCC(CNC(=O)CCc2ccsc2)N(C(c2ccc(Cl)o2)=O)C1 c1(C(N(CC(C)NC(c2cc(C)cc(Cl)c2)=O)C)=O)ccc(F)c(Cl)c1N C1(NC(Cc2c(C)noc2)=O)CCN(C(=O)CC2(C#N)CC2)CC1O c1(N(C2CCN(C(c3cccc4ccnn34)=O)C2)C)ncc2c(n1)CCCCC2 c1(SCC(=O)NC2C=CC(NC(=O)CC(O)CC3CC3)C2)nc2ccccc2s1 N1(C(CN(C)CC)=O)CCCN(C(c2ccc(C(C)C)c(C)c2)=O)CC1C(C)C CCC(C)(C)C(O)C(=O)N1CCC(OCC=CCNC(=O)OC(C)(C)C)C1 c1(C(N2CC(OCC)C(CNC(c3cc(C)no3)=O)C2)=O)nc(C)ccc1O C(=O)(CC(O)C(C)C)NC(CCC(=O)NC1CN(CC)C(=O)C1)C c1(C(=O)NC2(COC)CCN(C(=O)CNS(C)(=O)=O)C2)ccc2c(c1)CN(C)C2 c1(OC)ccnc(CNC(c2ccc(CNC(=O)CC3C=NN(C)C3=O)cn2)=O)c1 CC(CN1CCOCC1)C(=O)NC1(CNC(=O)CC2CC23CC3)CC1 N1(C(C2C(=C)C2)=O)C2CCCC1CN(C(c1c(OC)ccnc1OC)=O)CC2 CS(=O)(=O)CCCC(=O)NC1(CF)CCN(C(=O)CCC2CCOCC2)C1 CC1(CN=c2[nH]nc(CO)s2)CCCN(C(C2CCCCCC2O)=O)C1 c1(C(=O)NC(CNC(C=Cc2n(CC)ccn2)=O)C)cc([N+](=O)[O-])c(C)s1 O=C1C(c2ccc(Br)cc2)CCN1CC(N1CCCC(N2CC3CCC2C3)C1)=O c1(CCC2(NC(=O)Cc3cccnc3)CN(C(C3CC3F)=O)C2)ccc(F)cc1 c1(N2CCC3(CC(NC(c4ccc[nH]4)=O)C3)C2)c(F)cc([N+](=O)[O-])cc1F c1(COCC)nc(N2CCC(C(C)NC(=O)CC3(C)CCCC3)C2)cc(C)n1 c1(C(N2CCC(C)C2CNC(c2cc(O)nn2C)=O)=O)cc2c(nn1)CCCO2 Cn1nnc2cc(N)sc12.N12CC(C(O)C1)C2=O.C1(OCCN)CCCCC1OC Cn1ccc(C(=O)NCC(CNC(c2ncccc2CO)=O)CO)cc1=O N1(C(Cc2c(CC)cccc2)=O)CCN(C(c2ccc(C)cc2)=O)C(CCO)C1 c1(C(=O)NCC(CC(C)C)NC(=O)C(Cl)=CCl)ccc2nnc(O)n2c1 CCC1=NOC(CC(=O)NC2CC(N(CC(=O)SC3CCCO3)C)C2)C1 C(C(C)(C(=O)N1CC=CC(O)C1)NC(c1ncsc1C)=O)SC c1(C(=O)NC2CN(C(c3cc[n+]([O-])cc3)=O)C2)cnc2c(Cl)cccn12 c1(C(=O)NC(C2(O)CN(C(CCC(=O)NC)=O)C2)C)cnc2c(c1)COCC2 C1(NC(C2CC2(F)F)=O)CCCCN(C(=O)Cc2csc(Cl)n2)C1 N1(C(C2(COC)CC2(F)F)=O)CC2CCCCN2c2ccccc21 C(C(=O)N1CCCc2nccn21)(C1CCOC1)NC(c1nocc1Cl)=O CC1=C(Br)CN(C(=O)C(CC(C)C)n2ccnc2)CC1 C1(NC(c2ncc(OCC)nc2)=O)CCCCN(C(=O)C2CC2)C1 N1(C(Cc2cc(C(C)=O)no2)=O)CCN(CC2CN(C(=O)CCCOC)C2)CC1 C1(C#CC(=O)NC(C)CNC(=O)C(C)(C)c2ccncc2)(CC)COC1 n1(CC(=O)NC2CN(C(c3n(C(C)C)cnc3)=O)C3C2C3)cnc([N+](=O)[O-])c1 c1(-c2cncc(CC(=O)Nc3ncc(OC)c(C)n3)c2)ccc(F)c(C)n1 C1(CC(=O)NCC2N(C(C(C)SC(C)C)=O)CC2)CCC(F)(F)CO1 c1(OC)ccccc1CNc1ccc(CC(=O)OCC(N)=O)cc1 c1(C(=O)NCC2C=CC(NC(c3c(OC)csc3)=O)C2)ccc2c(c1)CN(C)CC2 N1(C(C2CC(C)CN(C(=O)C3=COCC3)C2)=O)Cc2cncnc2C1 C1(NC(c2cccc(OC)c2)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)C(C)C1 C1(CCNC(CCOC(C)C)=O)CSCCN1C(=O)Cc1coc(C(F)F)n1 c1(CNC(=O)NC2CCC(NCc3c(C)cccc3)C2)nc(Cl)ccc1Cl N1(C(c2c(C)cn(C)n2)=O)CCC2(CCN(C(c3cc4ccccn4n3)=O)C2)C1 c1(C(=O)NC(CN(C(Cn2c(C)cnc2)=O)C)C)cc(O)cnc1N C1(NC(C(=O)NCCOC)=O)CCC2CN(C(c3csc4cncn34)=O)CC2C1 c1(CC(=O)NC2CN(C(C(COC)OC)=O)CC2(C)C)cnc2c(C)cccn12 C#CC1(O)CCCN(C(=O)C(F)(CNC(C2(SC)CC2)=O)C(C)C)C1 C=CCC(C)(C)CC(=O)NCC1CCCC1NC(=O)Cc1cccc(F)c1O c1(C(=O)NCCC=C)ccc2c(Nc3c(C)noc3C)n[nH]c2c1 Cc1cc(C(N)=O)c(NC(=O)CC2CCN(C(=O)NC3C=CC(=O)N=N3)CC2)s1 CS(=O)C=CC(=O)NC(Cn1cc(C(=O)O)cn1)C(=O)O c1(CN(C(=O)CC2C=CC(NC(=O)C(F)C(F)(F)F)C2)C)ccc2c(c1)CCO2 N#Cc1nc(-n2cnc(-c3nc(C4CC4)no3)c2)n[nH]1 C(=O)(C(CCC1CCC1)NC(c1nonc1N)=O)NCC(c1ccsc1)C Cc1sc2ncc(C(=O)NC3CCCCC3n3cccn3)n2c1C Cc1cc(C)n(CC(=O)NC(C)CCCCNC(c2cc(C(C)C)[nH]c2C)=O)n1 O=C(CCNC1CC1(C(F)(F)F)CO)N=c1nc(-c2ccccc2)[nH]s1 N1(C(c2c(OC)ccs2)=O)CCN(C(=O)CC2(C)CC(C)=NO2)CC1C c1(C(N2CCCC(NC(c3c(C)ncc(N)c3)=O)C2)=O)cc(S(N)(=O)=O)co1 C#CC1(NC(=O)CC2CCCC2NC(=O)C(C)(C)Cl)CCC(C)(C)C1 c1(C(C)C)cnc(O)c(C(=O)NC(C)(CNC(=O)CCC=CBr)C2CC2)c1 N1(C(c2c(CCCC)ocn2)=O)CC2(CC(NC(c3cnncc3O)=O)C2)C1 c1(C(N2CC(NC(c3c(C)n(C)nc3)=O)CC2(C)C)=O)cc2cc(O)ccc2[nH]1 c1(NC(C(CO)NC(c2cc(C)cc(O)n2)=O)=O)cccc(C#N)c1C N1(C(c2c(C(C)C)ncs2)=O)CC(NC(C2CC(C)(C)C2)=O)C(C2CC2)C1 Cc1ccc(C(=O)NCC2(O)CCN(C(=O)Cc3nncn3C)C2)nc1O C1(C)(C(N2CC=CC(NC(c3cc(C)oc3)=O)C2)=O)CCCCC1(F)F c1(C(N2C(C)(C(N(C3CCN(C)C3)CC)=O)CC2)=O)ccc(CO)cn1 c1(CC(=O)NCC(N2CCCC2CC2CC2)=O)cnc(C2CCC2)s1 C1(CNC(c2cccc(C)c2)=O)CCCC2(CN(c3nnc(C(N)=O)s3)C2)O1 c1(OC)ccc(Br)c(F)c1CN1CCn2ncnc2C1 c1(N(C(N(C(C2CCCO2)C)C)=O)C2CC2)cccc(-c2nccs2)c1 N1(CC=CC(=O)NCC2CC2)CCC(C(N(C2CC2(F)F)CC=C)=O)C1 C1(NC(=O)CC2OCCO2)CC2CCC1N2C(c1c(Cl)nsc1Cl)=O CCCCCC(F)C(=O)N1CCC(NC(c2cc(C)on2)=O)C(C(N)=O)C1 C1(NCc2nnc(C)s2)CC(NC(=O)CCN2CCCCC2)C12CCC2 N1(C(c2c(CC)onc2)=O)CCN(C(C)CNC(=O)C(C)(COC)OC)CC1 CC(CC(=O)N1CCC(CC(=O)NCCn2cccc2)C1)C(F)F Cc1ccncc1CN(C(=O)CC(C)N(C)C)C.C1(=O)C(C)CN1 c1(C(C(=O)NCC(CN(C)C(c2cn(C3CC3)cn2)=O)O)(C)C)ccccc1F c1(SCC(=O)Nc2cc(C)nn2Cc2ccc(Br)cc2)ccc(F)c(F)c1 N1(C(C=CCC)=O)CC2(C1)CN(C(c1c(F)cc(O)cc1F)=O)CC2CO CCCN=C(NCc1cccc(OC)c1OC)Nc1ccc(C2COC2)cc1 c1(OC)cc(C)ccc1NC(=O)C(C1CCCC1)N(C)Cc1ccn(C)n1 c1(C(N(CC(CNC(C(F)OC)=O)C)C)=O)ccc(C(N)=O)c(Cl)c1 N1(C(C2(NC(c3nccn3C)=O)C(C)CCC2)=O)CC=C(CO)CC1 C(=O)(CC(F)(F)CC(=O)N1CCCC(NC(c2cccc(CO)c2)=O)C1C)OC C1(O)(CNC(c2ccncc2C(F)(F)F)=O)CCCN(C(c2ccon2)=O)C1 c1(C(N2CCC(C3N(c4nnc(C)s4)CCC3)C2)=O)nn(C)c(Cl)c1Cl c1(C(c2cn(CCCC(=O)NC)nn2)(C)C)ccc(C(F)(F)F)cc1Cl c1(C(N2C(CC)C=CC2)=O)ccc(CF)cc1.C12(CC1)C(=O)N2.C(=O)(C1CC1)N CC1CCC(C(=O)NCc2cccc(C#N)n2)N(C(c2nn(C)cc2Cl)=O)C1 c1(CC(=O)NC2(C)CN(C(c3cc(CC)no3)=O)C2)ccc2nsnc2c1 C1(C)(C(=O)NC)CCN(C(c2sccc2Cl)C(=O)NC2CCC2)CC1 N1(C(c2c(CNC(CCN(CC)CC)=O)c[nH]n2)=O)CC2C3CCC(C3)C12 CC=C=CCCN=C(NCc1csc(C(F)(F)F)c1)NCC(C)C N1(C(c2ccc(F)s2)=O)CCOC2(C1)C1CC3CC(C1)CC2C3 C1(NC(C=CCN(C)CC)=O)C2CC(NC(=O)C(c3c(C)noc3C)C)CC12 C1(C(N(CCNC(CSCC=C)=O)CC2CCC2)=O)CCCC(C)(C)CC1 CCC(F)(F)CC(=O)N1CC(C(=O)NC(C)(COC)CCO)(COC)C1 C(CC(=O)NCC1(CO)CCN(C(C2(C)CC2)=O)CC1)(C(F)(F)F)N(C)C O=C1CC(C(=O)N2CCC(CC(=O)NCc3ccc(O)cc3)C2)=NN1 c1(C(=O)NCC2(C)CCCN(C(C3(C#N)CC(=O)C3)=O)C2)nnn2ccccc12 C=CCCCCCC(=O)NCCCCC1(NC(=O)C(F)CCC)CC1 c1(OC)cc(OC)c2cc(NC(c3ccc(C)s3)=O)[nH]c2c1 C1(CNC(CCC(=O)OC)=O)CN(C)CCN1C(C1CCN(C)C1C)=O N1(C(Cc2nc(C)sc2)=O)CC(NC(c2c(C(F)F)cccc2F)=O)CC(C)C1 O=C(C1=CC2(CCOC2)C1)NC1CCN(C(C2CCC3(C2)CC3(F)F)=O)C1 FCCCN=C(NCc1ccc(Cl)cc1)NC1CC(OCc2ccc(CO)s2)C1 C1(C(=O)NCCC2N(C(CCOCCOC)=O)CCSC2)CCN(C)C(C)C1 C(=O)(C(C)C(C)NC(C1CCO1)=O)NCc1nc(CC)[nH]n1 c1(C2(CC(=O)NC3N4CCC43)CC2)ccccc1.C1(OC)CC(CCC(C)C)C1 c1(SC)cccc(C(=O)NCC2CCC2NC(=O)C=CC(F)(F)F)c1 C(CCCC(CO)NC(=O)CC1CCC(C)(C)CC1)NC(Cn1ccc(C)n1)=O N1(C(c2nn[nH]n2)C)CCCN(Cc2ccc(SC(F)(F)F)cc2)CC1 c1(NC(c2c(NCc3cccc(OCC=C)c3)ccs2)=O)cnc(F)cc1C C1(C(N(CCN(C(C2CC(C(F)(F)F)(OC)C2)=O)C)C)=O)COC2(CCC2)C1 c1(C(=O)NC(C2(O)CN(C(c3cnn(CC)n3)=O)C2)C)ccc(OC)nc1 c1(C(=O)NCC23CCC(CC2NC(C24CC(F)(C2)C4)=O)C3)cc2cc[nH]c2cn1 c1(CNC(=O)NCCCc2ccc(Cl)cc2)nc2c(Cl)ccnc2[nH]1 C(=O)(C(CC(C)C)NC(=O)CCNC(=O)C1CC1)NC(C(=O)NC)(C)C CC1CN(c2ccnc(N3CC4(CCOC4=O)C3)n2)C(C)(C)CO1 c1(C(=O)OCC)c[nH]c(=NCC2(C)CCN(C(=O)C(C(C)C)N(C)C)C2)s1 Nc1c(Cl)cc(C(N2CC(NC(=O)C(F)(F)F)C3CC23)=O)cc1[N+](=O)[O-] N1(C(C(C)(C)OCC)=O)CCC(NC(=O)CCOc2ccccc2C)C(C)C1 C1(C(=O)OCC)CCN(C(=O)CCNC(=O)C(F)OC(F)(F)F)CC1 c1(OCCC(=O)Nc2ccc(NCC)cc2)cc(C)ccc1OC C(=O)(C(O)C(F)(F)F)NCCC1CC(C(=O)NC2CCC(COC)CC2)C1 C(N=C(NCC1CCCS1)NCC(F)F)C1(C#N)CCC1 Cc1cc(C(N2CCC(CNC(=O)Cc3ccnnc3)C(C)C2)=O)cc(C)c1F N1(C(C(=O)NCCCOC)C)CCCN(C(c2cc3ncccn3n2)=O)C(C)C1 C(C)(N=c1ccnc(NCc2csc(-c3ccccc3)n2)[nH]1)c1c(CC)nns1 c1(SC(C(C)C)C(C)NC(=O)Cc2cnccc2Cl)ccc2ccccc2c1 c1(CC(C(=O)N(CC(C)NC(=O)CC(C)F)C)OC)ccc(F)cc1 N1(C(C(C)OCCC=C)=O)CC2CC(N(C(C3(CC=C)COC3)=O)C3CC3)CC2C1 c1(C(C(=O)NC(CN(C(C23CC(C)(C2)C3)=O)CC)C)OC)ccccc1F C1(C(N(C2CCS(=O)(=O)C2)CC)=O)CCCCN1CC(=O)NC1CC2C=CC1C2 c1(OC)cc(C)sc1C(=O)NC1CCC(n2cc(C3CCCCO3)nn2)CC1 Nc1cc(C(=O)NNC2C3CN(C(=O)CC(=O)NC4CC4)CC23)ccc1F C1(NC(CNC(COC)=O)=O)CCC1NC(=O)C(c1ccoc1)SC CCC(C)(O)C(=O)NC(C)(C)CCC1CCCCN1C(=O)CS(=O)(=O)N(C)C S(=O)(=O)(c1cnnc(O)c1Br)Nc1ccc(OCCCC)c(C)c1 n1(CC)nc(C(=O)NCCC2CCCN(C(c3ccncc3)=O)C2)c(Br)n1 C1(C(N(CCc2ccc(OC)cc2)C2CC2)=O)Cc2ncccc2N1C(C)C c1(NC(c2nc(C)n(C)c2C)c2n(CC)nnn2)nc2cnccc2[nH]1 N1(C(c2c(C)n[nH]c2C)=O)C2CCC1CN(C(=O)C(C)CSC(F)(F)F)CC2 N1(c2ncc(C)cn2)CCC(O)C(c2nc(C(=O)NC(C)C)no2)C1.C(C)(C)(C)S C1(NC(Cc2cccc(C)c2)=O)CC(O)CN(C(c2cnccc2C)=O)C1 C(=O)(C1=CCCCC1C)NCCC1CC(C(=O)NC(C(=O)OC)(C)C2CC2)C1 N1(C(Cn2cc(-c3cccc(C)c3C)nn2)=O)CCC(O)C(C)(C)C1 C1(NC(C(CC)NC(C)=O)=O)(CO)CCN(C(=O)CC(C)(C)SC)C1 c1(CN(C(C)CNC(=O)Cn2cnnn2)C)cn(C)nn1 c1(CN(C(=O)CCC2(C)CC2)C)cccc(CNC(=O)C(C)(C)c2cnco2)c1 c1(CN(CCC)CC)cn(CC2(C(F)F)CC2)nn1.c1(C=O)cocn1 C(=O)(C(C)(O)CC(C)C)NC(CNC(c1cc(C)c(O)cc1)=O)C c1(C(=O)NCCCCCNC(c2c(SC)csc2)=O)cccc2ccc(C)nc12 Nc1ccc(C(=O)NCC2(C(=O)NCC3CC3CO)CCCC2)nc1 n1(CC)nnc(C)c1C(N1CC=CC(NC(=O)CNC(=O)C(C)(C)C)C1)=O N1(C(c2c(C)ocn2)=O)CCC(C(=O)NOCCOCCC2CC2)CC1(C)C c1(C(N2C(C)C(NC(C3CC3F)=O)CCC2)=O)cccn2c(CO)nnc12 Cc1nn(C)c(C)c1CC(C)C(=O)NCC(C(C)C)NC(C1(CF)CCC1)=O C1(CNC(CCCSC(C)(C)C)=O)CCCCN1C(C1CNC(=O)C1)=O C1(NC(CC2N(C(C(C(C)C)OCC)=O)CCCC2)=O)CC2CC1CC21CC1 c1(C(=O)NCC2CC(OC)CN2C(c2cc(C)cc(F)c2)=O)c(C)cncc1F c1(-c2ccc(OC)cc2C)cc(C)c(S(=O)(=O)NCC(F)CO)cc1C c1(OC)ccc2nc(N3CCCC(NC(=O)CC(F)(F)F)C3C)sc2c1 Cc1nc(F)ccc1-c1cn(C2CCCC2NC(C2(CC3CC3)CCC2)=O)nn1 c1(NC(C=CCNC(c2c(CC)ccs2)=O)=O)ccc(C)c(F)c1F c1(C(=O)NC2C(CNC(CCSCCCC)=O)CC2)cnccc1N(C)C C(C(CNC(=O)Cc1cc(Cl)ccc1Cl)C(F)(F)F)NC(C(C=C)(C)C)=O C(=O)(CCC(F)(F)F)NCc1ccc(C(N(C)CC2CCC(=O)N2)=O)s1 C(=O)(CCCCCC#N)N(CC(CC)NC(c1c(C)nn(CC)c1C)=O)C Cc1cc(Br)sc1C(=O)O.C1(=O)NNC(=O)N(C)C12CCOC2 c1(CC)conc1CC(N1CC(C(C(=O)NC(C)C(C)C)OC)C1)=O c1(C(=O)NC2C(N(C(C(=O)N(C)C)=O)C)CCCC2)cnc(O)cc1C(F)(F)F CS(=O)(=O)C1CCN(C(C2CC3CC3N2C(c2cc(Cl)ccn2)=O)=O)CC1 C1(CNC(CN(C(=O)CN2CCC(C)(C)C2)C)=O)CC2CCC1C2 C(=O)(C(C)(F)C(F)(F)F)NC(C)CC1CN(C(c2csc(-c3cnn(C)c3)n2)=O)C1 c1(C(=O)NC2C(CC)N(C(C3CCCC3)=O)CC2)ccc2c(n1)OCC(=O)N2 c1(N2CC(CNC(C(CC#C)(C)C)=O)OCC2)nc(C)nc2c(C)csc12 c1(C(C)=O)cccc(OC(C)C(=O)NC(C(=O)NCCCCCC(C)C)=O)c1 CC1(CNC(=O)C(=Cc2cccnc2)F)CCCC1NC(=O)CC(Cl)Cl c1(CCC(=O)NCC2CCN(C(=O)C3=CCSC3)C2)ccc(Cl)cc1F c1(C(=O)NC(CN(C(=O)Cc2ccc(O)cc2)C)(C)C)cnn2ccccc12 C(=O)(N=c1cc(C)o[nH]1)C12CN(C(C(CC)Sc3ccccc3)=O)CC1C2 CCC(C)C(C)(O)CNC(=O)CCN(C(c1c[nH]c(C)c1)=O)CC1CC1 c1(C(C)(C)OC)noc(C2(C)CC2(C)C)n1 C1(CCNC(CC(=C)C)=O)C(C)CCCN1C(=O)COCC(=C)C c1(C(=O)NC2(C)CC(NC(CSCCC)=O)C2)c(F)cc(Cl)cc1F N1(C(c2cc(OC)n[nH]2)=O)C2CCC1CN(C(c1cc3n(n1)CCCC3)=O)C2 C(=O)(CC(N=c1ccc(Br)c(S(=O)(=O)NCc2ocnc2C)[nH]1)C1CC1)NC C(=O)(C1=NN(C)C(=O)CC1)NC1C(CNC(c2cc(C)nnc2)=O)CCCC1 c1(C(=O)NC2(C)CCN(C(c3c(CC)nco3)=O)C2)cn(C)ccc1=O Cc1cccc(OCC(N2CCOC(Cn3cc(C4CCC4)nn3)CC2)=O)c1C C1(C(N2CC3(CN(C(CC4CCC(=O)NC4)=O)C3)C2)=O)CCC2C(C1)C2(F)F Cc1cccn2ncc(C(=O)NC3CC(NC(=O)CC4CC5CC5C4)C3)c12 Cc1sc(C)c(C(N2CC(NC(C3CC4CCC3O4)=O)CC(F)C2)=O)c1C#N c1(C(=O)OC)cc(N(C)CCc2cccs2)c2ccncc2n1 N1(C(C2(c3ccc(OC)nc3)CCC2)=O)CCCCC12CCC2 N1(C(CC2(N(C)C)COC2)=O)C2CCC1CN(C(C1CCS(=O)(=O)N1)=O)C2 Cc1ncccc1CC(=O)NC1CN(C(c2cn(C)nc2C)=O)CC1C(F)(F)F c1(C(N(C(C)C(=O)NC(C2(CO)CC2)C)CC)=O)ncccc1F C1(C)(C(N(CCN(C(C)C)C(c2cnnn2C)=O)C)=O)CCCN(C)C1 C1(OC)CC(NC(C23CCCN2CCC3)=O)CN(C(c2cncc(N)c2)=O)C1 c1(C(C)C)ccc(C(N2CCC(OCCNC(C3(C)CCCO3)=O)C2)=O)c(F)c1 Cc1ccc(C(N2CC(NC(=O)COCC3CCC3)CC(F)C2)=O)c(F)c1F c1(C(N2CC(C)(NC(=O)CC3C=CCC3)C2)=O)[nH][nH]c(=N)c1Br Cc1cnc(C(N2CCCCCC2CNC(=O)CCC2CCOC2)=O)cc1C#N N1(C(COC(C)(C)C(F)(F)F)=O)CC(F)(F)CC1CNC(C1CC1(C)C)=O N1(C(C2C(CCC)CN(C(=O)CC3(C)OCCO3)C2)=O)CCC2(CCCC2)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(C2CCN(C(N)=O)CC2)=O)CC(C)C1 c1(C(C)=O)ncnc2c1ccn2CC(=O)NC1(C)CN(C(=O)C(C)C(C)O)C1 C1(SCC)OC2CCC1CC2.O=C1CCCC2(CCC2)N1.c1(C)cn(CCCO)nn1 C(=O)(CCCCCC#N)NC(C(C)NC(CCC(=C)Br)=O)(C)C Cc1ccc(Br)c(CC(=O)OC(C)(C)C)c1.C12(CCN(C(N)=O)C1)CN(C)C2 c1(C(C(N2C(C(C)NC(C)=O)CCC2)=O)C)ccc(N(C)C)cc1 c1(CC(N2CCCC(NC(CSCC)=O)(CO)C2)=O)cccc2nonc12 C(C(CC)(CC)C(=O)NC1CC(O)C(O)C1)NC(c1ncc(CC)cn1)=O c1(C(N2CC(C)C(CNC(=O)CCc3ccncn3)C2)=O)c(F)ccnc1F C1(NC(C(C)O)=O)CN(C(c2cc(Cl)cc(Cl)c2O)=O)CC2(CCOCC2)C1 C(=O)(CC(C)C(C)C)NCC(CCOC)NC(c1ccc(N(C)C)nc1)=O c1(NC(c2n(SCC)c(O)nc2)=O)ccnc(OC)c1I C(C(C)C(F)C(=O)NC1(CCOC)CCCC1)NC(COCCCOC)=O c1(CC(=O)N(C2(C(N3CCC(CCC#C)C3)=O)CC2)C)ccc(C)cc1 C1(CC)C(C(=O)N(C)CCn2ccnc2C)CCN1C(=O)CN1CCC(OC)C1 c1(C(N2CCC(CCSCC)C2)COC)ccccn1.N(C)C N1(C(C2CCN(C)C2=O)=O)CCC(O)C(NC(C2(Cc3cnn[nH]3)CCCC2)=O)C1 C(=O)(C(C(=O)OCC)C(C)C)NCC(C)N(C(C(C=C)(C)O)=O)C O=C1CCC(CNC(=O)CN(C2CCC2)C(c2ccn(C3CC3)n2)=O)N1 N1(C(c2cc(C)[nH]n2)=O)CCCC12CCN(C(c1c(C(F)(F)F)coc1C)=O)C2 N1(C(=O)Nc2c(C(C)C)cccc2)CC2(C)CC1(C)CO2.c12ccccc1NC2 C1(CNC(C(CC(C)C)OC)=O)CC2CCCC2N1C(c1n[nH]cc1F)=O C1(C(C(=O)N(CCC(N)=O)CC)(C)C)CCCN(C(=O)CC(C)C)C1 c1(-n2cc(C3N(C)CCN(C(C=CC=CC)=O)C3)nn2)cccc([N+](=O)[O-])c1 Cc1cccc2cc(C(N3CCC4CN(C(C5CSCCS5)=O)CC34)=O)oc12 c1(NCC2C(NC(CCC(C)SC)=O)CCC(C)(C)C2)cccc(F)c1[N+](=O)[O-] Cc1cc(C(=O)NCC(CC(F)(F)F)NC(c2sncc2C)=O)c(Cl)cn1 c1(C(=O)NCCN(C(=O)COCc2ccco2)CC)cc(C)nn1-c1ccccn1 N1CCc2cccc(O)c21.CC1CC(F)CN1C C1(CO)CC2(CCCCCC2)C1.c1(C2CN(CC)C(=O)N2)cccc(Cl)c1 N1(C(c2cc(C)on2)=O)CC(NC(=O)Cc2ccc(OC(C)C)cc2)C(O)C1 C12(C(=O)NC3CN(C(c4cc(C)on4)=O)CC3C)CCC(N=[N+]=[N-])C1C2 c1(OC)cc(C(=O)NCCCN(C(=O)CC2CC3CC3C2)C)cc(F)n1 C(=O)(CCCC(F)(F)CO)NC(CCCCNC(C(C)C(F)F)=O)CO O=C1CC(C(=O)N2CCC(CCNC(C3CCCS3(=O)=O)=O)C2)c2ccccc21 CCS(=O)(=O)CC(=O)N1CCOCC(NC(c2cccnn2)=O)C1 C1(NC(c2c(CC)scc2)=O)CCOC2(CCN(C(=O)COC(C)C)CC2)C1 c1(C(N2CC(F)(CNC(C3C(C)(C)CC3)=O)C2)=O)ncn2cc(Br)sc12 c1(C(=O)NC(C(C)NC(C(COCC)(C)C)=O)C)ccc(OC)c(F)c1 c1(OC)ccccc1CNC(c1nnnn1C1COC1)C1CC1.c1(C)ccon1 c1(C(=O)NC(C)(C)CCNC(=O)CC2C=CCCC2)cnc2c(c1)NCC2 C1(O)(CC=C)CCN(C(C2(F)CC(NC(=O)C(C)N=[N+]=[N-])C2)=O)CC1 c1(NC(C2N(C(CC(C)C)=O)CCSC2)=O)cnc2[nH]cnc2c1 n1(CC(=O)NCCC2(O)CCN(C(C3CCCCO3)=O)C2)cnc2c1CCCC2 C1(CCC=C)(C(=O)NCC(F)=C(C)C)CN(C(=O)C(C2CCCCC2)O)C1 N12CCN(CC1)C(=O)CCCN1CCN(CC1)CCC(O)C2=O.C(C)(=O)N.CCO C(=O)(CCCS(C)(=O)=O)N(C1CC(C(N2CCCCC2C2CCCCC2)=O)C1)C C1(CCNC(C2C3CCC23)=O)CCCCN1C(C1(F)CCCC1)=O N1(C(C2C(CCOC)C2)=O)CC(CNC(c2cc(Cl)c(C)cn2)=O)C2(CC2)C1 C1(CCNC(c2c(C)[nH]cc2)=O)CC(F)(F)CN1C(=O)CNc1cccc(F)c1 C1(NC(C2CCCC(F)C2)=O)CCCCC1Nc1ccc(C(F)(F)F)cn1 N#Cc1ncc(N2CC3CCC2CN3C(=O)C(O)Cc2ccccc2)nc1C#N C1(NC(c2cn(CCOC)nc2)=O)CC2CCC(C1)N2C(=O)CCOC1COC1 C#Cc1ccc(C(=O)N(CCCNC(c2nn(C)cc2C)=O)CC)c(F)c1 C(=O)(C(C(C)CC)N(C)C)N1CCN(CC(=O)N(CCCF)CC#C)CC1 Cn1nnc2c1CCN(C(C13CC1CN(C(c1cc4ncccn4n1)=O)C3)=O)C2 Cc1nn(CC(F)(F)F)c(=O)n1C(c1ccccc1Cl)C CC1CN2CCN1C(C(=O)NCC1C3N(C(=O)COCC4CCC4)C(CC3)C1)C2 N1(C(C=C(COC)C)=O)CC2CCCC(C1)N2C(C1CCn2ccnc2C1)=O CCC(C)CCC(O)CC(=O)N1CCC(NC(C2CCSCC2)=O)C1 c1(C(=O)NCC2CN(C(c3[nH]c(=N)sc3)=O)CC2(F)F)cc2nc[nH]c2cc1F C1(C(N2C(C(=O)NC(C)(C)C)CC(OC)C2)=O)CC12CCSCC2 C(CCN=C(NCCC1CCC1C(F)(F)F)NC1CCS(=O)(=O)C1)OCC c1(SCC)nccnc1C(=O)N(C1CN(C(=O)C=Cc2ccnn2C)C1)CCO c1(C(=O)NC2CCCN(C(CC3C(=O)NC(=O)N3)=O)C2)cn2ccnc2cn1 Cc1cc(-c2ncco2)ccc1NCc1cnc(C2CCOCC2)o1 c1(CC(=O)NCCC2(CNC(C(CCC)=CCC)=O)CC2)ccccc1[N+](=O)[O-] C1(CN(C(C2(C)C(C)C2)=O)C)CCCN1C(=O)C=C1CCSCC1 C(=O)(CC(C)C(F)F)N1C(CN(C(c2nn(CC)c(C)c2)=O)C)CCC1 C1(CC(=O)N(CCCCNC(=O)C(C)(C)c2ccsc2)C)CN2CCC1CC2 C1(CC(=O)N(CCCNC(CC=CC)=O)C)CCCCN1C N1(C(CCOC)=O)CC=C(C(=O)NC(C)CC2CCC2)C1 C1(OC)CN(C(=O)CCCCF)CC1NC(C1CCOC(C)C1)=O C1(N(C(C2(CCOCC)CCC2)=O)CCO)CCN(C(=O)C(C)=C2CCCC2)C1 C=C(F)C1(CC(=O)NC2(C(=O)NCCCN3CCCC3=O)CC2C)CCC1 c1(C(N2C(CNC(c3n(CC)c(O)nc3)=O)CCC2)=O)cnc2c(C)cnn2c1 N1(C(C(=O)NC)C(c2ccccc2)OC)CCOC2(CCN(C)CC2)C1 C1(CCC(C)C)CN(C(=O)C(=O)NCC2CCCN2c2ccccc2)CCO1 c1(C(=O)NCCCCNC(CCc2ncc(C)[nH]2)=O)cn(C)nc1O N1(C(=O)NC(N(OC(CCC)C)Cl)=O)CCN(C(CC(C)C)=O)CC1 C=C(C)C1OCCC1C(=O)NC1CN(C(=O)C=Cc2ccccn2)CCC1F C(=O)(C(O)CSC)N1CC(OCC(=O)NC(COC)CO)C1.C(CF)O N1(C(C#CC(C)(C)O)=O)CCC2(C1)CN(C(c1ccnc(C3CCCC3)n1)=O)C2 Fc1ccc(-n2nc(C3C4COCC34)nc2-c2cc3ncccc3[nH]2)c(F)c1F N1(C(c2c(CCC)nns2)=O)CCC(C)C1CNC(=O)CC1CSCCS1 C(=O)(C(=O)C(C)(C)C)NCC(C(N1CCC(N(C)CC)C1)=O)C CCCC(C(C(=O)NCCOC1CC1)N1CC(c2ccc(C)cc2)CC1C)OC CC1C(C)N(C(c2ccc(C(N)=O)[nH]2)=O)CCN1C(c1cc2n(n1)CCC2)=O C1(C(C)NC(COC(CC)(C)C)=O)CCN(C(c2ccn(C(C)C)n2)=O)C1 CC1=NN(C)C(=O)C1CC(=O)NC1CC(CNC(C2CCSCC2)=O)C1 C1(CNC(c2c(C(=O)NC(c3ccccc3)C)cccc2)=O)CCC2(CC2)CO1 c1(C(C(=O)NCC(CO)NC(C=CC=CCCCCC)=O)C)ccc(F)cc1F C1(C(=O)O)CC2(CCC(CNC(C(F)(F)C(F)(F)F)c3ccccc3)CC2)C1 c1(C(CC)C(=O)OC(C)(C)C)cc(C(F)(F)F)cc(Br)c1.C1(=O)COC(=O)N1 CC1CCCC1(C(=O)NOCCN(C)C)NC(c1cccc(SC(C)(C)C)c1)=O CC(C)CC(O)C(=O)N1CCC(NC(=O)CCOc2ccc(F)c(F)c2)C1 C(C(CC(=O)NCCCCCF)NC(=O)COCC1CCCCO1)OC C1(C(N(CCCC#C)CCNC(=O)CCc2ccsc2)=O)CCCCC1NC C1(NC(CCc2cc(OC)no2)=O)CCN(C(=O)CCc2cc(C)cs2)CC1C C1(c2n(C)cnc2)C(=O)NCCN1S(=O)(=O)CC1CCC2(CC1)CC2 C(=O)(C(C)CC(=O)NC1CC2CC(NC(c3cc(Cl)cs3)=O)CC12)OC C1(NC(CC2C(C)C2)=O)CCSC12CN(C(C1C3CCCCCCC13)=O)C2 c1(C(=O)NC(CC)(CNC(C2(S(C)(=O)=O)CC2)=O)CC)coc2cc(C)ccc12 c1(CC(=O)NC(C(C)NC(C(C)=CC)=O)(C)C)csc2cc(Cl)ccc12 c1(C(=O)NC(C)C(C)NC(=O)C(C)OCc2ccccc2)cccnc1C(F)F N1(c2nc(C)nc(C)c2F)CCC2(CCCC2NC(=O)C(O)CCC(C)C)CC1 C1(C(=O)NCC2CC(NC(c3ccc(C)o3)=O)CC2O)CC12CC(C)(C)C2 C1(NC(C(C)Oc2cccc(O)c2)=O)CN(C(C2(C)CC=CCC2)=O)CC1(C)C c1(C)ccccc1O.N1(c2ccnc(OC(C)C)n2)CCC(CO)(CO)CC1 c1(C(=O)NC2(CN(C)C(C3CC3C(F)F)=O)CC2)cnc2nccn2c1 N1(C(Cc2ccn(C)n2)=O)CC(C(N2CCC(CC3CCC3)C2)=O)C(F)(F)C1 N1(C(C2(C)CC=CC2)=O)CC2CCC2(CC(=O)NCC2(C)CCCCC2)C1 C1(NC(CC2CC(NS(C)(=O)=O)C2)=O)(CO)CCCCCC1.n1(CCCN)ccnc1 Cc1c[nH]cc(C(=O)NCC(C)CN(C(=O)CCCCN(C)C(C)C)C)c1=O C1(C(N2CCC(=CCNC(C3C(OC)CCC3)=O)CC2)=O)CCc2nncn2C1 c1(C(N)=O)cc(C(N2CCC(CNC(=O)C[SH](c3ccsc3)CCN)C2)=O)ccn1 C1(C(NOCCCOC)=O)(CN)CC12CCC2 N1(C(=O)NCCCOCCCOC)CCCCC1C1=NCCN1 O=C(C1=NOCC1)N1CC=CCC1C(=O)NC12CC1CNC2=O c1(C(C)NC(c2c(CNC(c3c(CC)c[nH]c3)=O)cc[nH]2)=O)cccc(O)c1 CC1=C(C(=O)NCc2cn(CCNC(C3CC(C4CCCC4)C3)=O)nn2)SCCO1 Cn1nc(C(=O)NCC2(C(=O)NCc3csnn3)CCCO2)ccc1=O N1(C(C2C(C)(C)C2)=O)CC2CC3CC2C1C3NC(c1nccn2nccc12)=O C12(CNC(C3C(C)(C)C3CNC(c3cnc(O)c(F)c3)=O)=O)CCC(CC1)CC2 Cc1noc(CC(=O)NC(C(=O)NCCN(C2CCCC2)C)c2cccs2)n1 Cc1n[nH]c(C)c1CC(=O)NC(C1CCCCC1)CNC(C1CC2CC12)=O Cc1cccnc1C=CC(N1CC(CN(C(=O)C=CBr)C)C2(CC2)C1)=O c1(OC)cc(Cl)c(S(=O)(=O)N2CCOC(C)C2CN)cc1Cl C1(CC(=O)NC(CN(C)C)CO)C2CCCC2N1C(=O)CCP(C)(C)=O C1(c2ccccc2)(CNC(CCCOC)=O)CCN(C(c2cnco2)=O)C1 C(=O)(CCCCCCNC(C)=O)NC(CNC(c1c[nH]c(=NC)o1)=O)C(C)(C)C C1(C)(C(=O)NCC(CCC)n2cccn2)CCCN(C(c2cnc(C)[nH]c2=N)=O)C1 N1(C(C)=O)CCC(O)(C2CCN(C(c3ccnc(C4CC4)c3C3COC3)=O)CC2)C1 N1(C(c2scc(OC)c2)=O)CCC(CF)(NC(=O)CC(C)c2ccco2)C1 N1(C(C2(C)CC2)=O)CC2CCC1C(NC(=O)CCC1(C)CCCCC1)C2 c1(CC)ccc(C(=O)NCCCCC(C)NC(c2cccs2)=O)cc1OC CC(CC(F)(F)F)C(=O)N1CCC2CC12C(=O)N(C1CC(O)C1)C C1(C(C)=O)C(C(=O)N(CC(=O)NCc2nncs2)C2CC2)C1(C)C c1(C(N2CC(CC=C)(NC(c3nncn3C)=O)C2)=O)occ(C)c1C c1(C(c2n(C(CC)C)nnn2)NC(C)(C)CSC)cccc2ccoc12 CCC(C)C(C)N=c1nc2sccc2c(N(C)Cc2c(F)ccc(Cl)c2F)[nH]1 Cc1ccc(C=CC(=O)NC(C2CCCC2)CNC(c2ccc(Cl)o2)=O)cc1 c1(C(=O)NC(CN(C(C(C)CN(C)C)=O)C)C)cc2c(Cl)c(F)ccc2[nH]1 C(C1(C)CCOCC1)=CC(=O)N(CCCNC(C1(COC)COC1)=O)C c1(C(=O)NC2CCCCC2(F)F)ccc2c(c1)CN(C(c1nc[nH]n1)=O)CC2 C1(NC(c2c(C)nncc2)=O)CCSC12CN(C(=O)C(F)(F)c1ccncc1)C2 N(C(=NCc1ccnn1C)N(C)CC1CC(SC)C1)CC(COC)(C)OC N1(C(C(CC(C)C)O)=O)CC2CC(NC(c3c[nH]nc3C3CCC3)=O)CC(C2)C1 C(=O)(NNC(=O)C(N)=O)Nc1cn(Cc2cccc(OC)c2OC)nn1 C#Cc1cccc(C(N2CCC3(NC(c4cc(N)c(Cl)cn4)=O)CC3C2)=O)c1 C(C(F)(C(=O)NCC(C1CC1)OC)C(C)C)NC(Cc1c(CC)con1)=O C(=O)(CCCCC(=O)N1CC(NC(c2c(CSC)cnn2C)=O)C(C)C1)NC C(C(CC(C)C)C(=O)NC(C)CC(C)NC(c1ccc(O)nc1C)=O)OC Cn1cc(CC(=O)NCC2(NC(=O)Cc3cscn3)CC2)nn1 c1(N(CCC(C)(C)C(F)(F)F)C)nccc(=NCCCCc2cnc[nH]2)[nH]1 c1(C(N2CC(N(C)C(c3c(F)ccc(O)c3F)=O)C2)=O)cc2c(cn1)COCC2 c1(C(=O)NC(C2CCN2CC)=O)ccc(CO)c(F)c1.c12cnn(C)c1NC2=O C1(C(=O)NCCCOCCNC(C2C(c3n(CC)ncc3)C2)=O)C(C#N)C1(C)C O=S(=O)(CCN=c1[nH]c2ccccc2s1)N1CCC(C(F)(F)F)CC1 C(=O)(C#CC1(C)CC1)N1C(C2CN(C(c3[nH]cc(C(C)(C)C)c3)=O)C2)COCC1 C#Cc1ccc(C(N2CC(CNC(c3ccc(F)c(C)n3)=O)C(C)C2)=O)cc1 C1(O)(CNc2ncc(C(=O)OCC)s2)CCN(C(=O)C(O)C2CC2)C1 C1(O)(CC(=O)N(C(C2C(C(N(CC(C)C)CCO)=O)C2)=O)C2CC2)CCCCC1 c1(C(=O)NCCC(CNC(CCCCOC)=O)O)c(N)ccc(F)c1C CCC(C)(COC)C(=O)NCCC(=O)NCC1CCCC12CC2 Cc1cnc2c(C(=O)NC3CC(NCc4ccc(C#N)nc4)C3)cnn2c1 C(CCN(C)C(c1cc(Cl)no1)=O)(C(C)C)NC(CCC=CC)=O C1(C(N2CCC(NC(CC(C(C)C)O)=O)(CF)C2)=O)CC2(C1)CC1(CCC1)C2 C1(O)(CN(C)C(c2ccns2)=O)CN(C(=O)CSC(F)(F)F)C1 c1(OC)cc(C)c(NS(C)(=O)=O)c(C)c1.c12cc(F)ccc1OCc1nnc-2o1 c1(C(=O)NC(CCCC)CNC(=O)C(O)CC(N)=O)cn(C)c(C)c(Br)c1=O O=C(C1=COCCO1)NC1CN(C(=O)CCc2ccccc2)CC2CC12 c1(NC(CCC)(C)c2nnnn2CC2CCOCC2)ccc2ncn(C)c2c1 C(CC(=O)NCCCC(C)(C)OC)(C(C)(C)C)NC(C=CC)=O CC1(C)CC1(C)C(=O)NC(c1ccccc1)CNC(C12CC(F)(C1)C2)=O c1(C(=O)NCC2CC(CNC(C3COC3)=O)CO2)cn2cccnc2n1 N1(CC)CCN(CC(=O)NCCCCNC(C2CCCC(=O)O2)=O)CC1 C1(S(C)(=O)=O)(C(=O)NCC(CCNC(CCC=CCC=C)=O)O)CCOCC1 C(=O)(C1CCCc2scnc21)N1CCC(O)(CCNC(CSCCC(C)C)=O)C1 c1(OCCCC(C)C)ccccc1C(N1CCCC(n2ccnc2)C1)=O Cc1c(C(=O)N(C2(C(=O)NCC3CN4CCC3C4)CCC2)C2CC2)cccc1F c1(CC(N2CC(NC(C3C(CCC)C3)=O)C2)=O)csc(-c2ncccn2)n1 c1(OC)ncc(C(=O)NC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C)nc1C C1(CCNC(c2c(CC)cno2)=O)CN(C(=O)C(F)CC2CC2)CCO1 C(C)(CCc1ccco1)(c1nnnn1CCSCC)CC(CO)OCC N1(C(CC2C(C)OCC2)=O)Cc2[nH]nc(C(=O)N(C3CC3)CC3CCCC3)c2C1 N12CCC(C(CO)C1)C2=O.c1(C(C)OCC)ccn(-c2ccccc2)n1 C1(NC(CN(C(C(C)OCC=C)=O)CC2CC2)=O)CCOC(C)C1 c1(NC)cnccc1C(=O)NC(C(=O)NC1CC1(C)C(N)=O)C1CCOC1 c1(NC(COC)C2CC2)ncc(C)cc1S(=O)(=O)NCc1ccc2c(c1)OCO2 N1(C(c2c(C)ccn2C)=O)CCN(C(=O)C(c2c(C)noc2C)C)C2COCC12 C1(C(=O)O)(C(=O)OC)CC1S(C)(=O)=O.n1(C(CC)CC)nc(C)cc1C(=O)N C1(O)(C(N(C2CCCC2)CCNC(C(C2CCC2)OC)=O)=O)CCOC1(C)C N1(C(C(c2cc(C)cc(C)c2)C)=O)CCOc2cc(C)c(Br)cc21 c1(C(=O)NC2CCC(NC(C3CCC(=O)NC3)=O)C2)cc(Br)cc(Cl)c1F C1(NC(Cn2ncc(C)c2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 Cn1cc(C(CO)NC(=O)NC2CCOCC2)c2ccccc12 C=CCCCCC(=O)NCC(CC(F)(F)F)NC(C1C2CCC(=O)C12)=O C(=O)(CCCCc1cccc(O)c1)NC1C(CNC(=O)C=CCO)CC1 n1(CC(=O)NC(CC)CNC(C2CCOC(C)C2)=O)ncc2ncccc12 N1(C(COCC)=O)CCC(C(=O)N(CC(C)C)CCO)CC1 C(N=c1ccc(Br)c(S(=O)(=O)NCC2(C)CSC2)[nH]1)c1c(Cl)ccc(OC)c1 C(CCCCC(=O)Nc1csc(C2CC2)c1)N(C)C(C1CC1F)=O c1(C(N(C2CN(C(c3cc(CCCCC)[nH]n3)=O)C2)C)=O)n[nH]c2c1COCC2 c1(C(=O)NCCN(C(=O)Cn2ccnn2)CCOC)sc(S(N)(=O)=O)cc1C c1(C(=O)NCCC(C)N(C)C(C2CNC(=O)N2)=O)cc2c(cc1O)OCO2 c1(CC(=O)NC2CCN(C(c3ncc(C)nc3)=O)CC2O)c(C)cc(C)nc1O C1(NC(CONC(Cn2c(C)ncc2)=O)=O)CC2CCC(C1)N2C(C)C C(=O)(CCC(C)(C)C#N)N(CCCOCCN(C(C(CC=C)(F)F)=O)C)C.C(CF)O C1(C(=O)NC(CCOCCNC(Cn2ncc(C)c2)=O)(C)C)CCC2CCC1O2 C1(CN(C(=O)C2=CCOC2)C)CCN(C(c2[nH]ccc2-c2cccs2)=O)CC1 N1(C(C(C=CC)O)=O)CCC(OC(N2CCCC2Cc2cccc(Cl)c2)=O)CC1 Cc1ccc(F)c(C(N2CCN(C(c3ccc(C)c(C)c3)=O)C3CC23)=O)n1 Nc1c(C(=O)NCC(O)CNC(=O)C=Cc2cscn2)sc2ncccc12 Cc1cc(C(C)C)ccc1C(=O)NCCOCCN(C)C(C1(C)CC1)=O c1(C(N2CCCC(NC(C(C)NC(C)=O)=O)CC2)=O)cc(C#N)cc(C)n1 Cn1cc(C(N2CCCCC2CCNC(C2CN3CCN2CC3)=O)=O)ccc1=O N1(C(C2N(C=O)CCC2)=O)CCCC2CN(C(=O)C(F)(F)c3cscn3)CC12 C(=O)(C(F)CC(C)(C)NC(=O)CN1CC2CC2C1)N(C(C1CCCO1)C)C C(=O)(CCNC(C1CN(C(N)=O)C1)=O)NC(C)Cc1ccco1 CC(C)C(O)C(=O)NC(c1ccccc1)Cc1ccc(F)cc1 c1(CNC2CCC(C(N3CC(CCC)C3)=O)OC2)ccc(S(C)(=O)=O)cc1C n1(CCC(C)C)c(NCc2ccc(OC(C)C)cc2Br)nc2ccccc12 C1(NC(C(C)(C)C2CC2)=O)CCN(C(=O)C=CSc2ccccc2)C1C1CC1 C1(CC)CN(C(=O)Cc2ccsn2)CCC1NC(=O)Cn1nc(C)c(Cl)c1C c1(C(=O)OCC)cccc(C(=O)NC2CC2C(=O)Nc2ccc(C(F)F)nc2)c1 CC1CC(C(=O)NCCC(O)CNC(c2cscc2C(F)F)=O)=NO1 C1(C(=O)NC(CCC)(C)C)(CC)CCCN1C(c1nonc1CC)=O CC(C(=O)NC1CN(C(=O)CC2CCC(C)(C)CC2)CCC1F)C(C)(C)C CC1COc2c(C(=O)NC(C)CN(C(=O)CCc3nccs3)C)cnn2C1 c1(N(C(C(C2CCCN(C(=O)CCC(=O)C3CC3)C2)C)=O)C)cccc(F)c1 C(C(=O)NCc1c[nH]nc1C(=O)N(C1CC(C)OC(C)C1)C)(C(C)(C)C)SC Cc1cnccc1CCNC(C1CC2(C1)CC2C(F)F)c1nnnn1CC(F)F C12(C(N3CCCC(CNC(CCC(=C)Cl)=O)C3)=O)CCCC1CC(=O)CC2 Cn1c(C(=O)Nc2cccc(C3CC3)c2)cc2ccccc12.C12CC1C(=O)NC2 C1(NC(=O)Cc2ccc(F)nc2)CC2CCC1N2C(=O)CC1CCOC1 C(c1nc2ccccc2s1)=CC(=O)NCCCCCNC(C1(NC(N)=O)CC1)=O c1(C(C)C)c[nH]nc1C(=O)N(C1CCC(NC(=O)CC(=O)N(C)C)C1)C CC1C(CC(=O)NCCOC(C)(C)CNC(=O)C(O)c2cnc[nH]2)CC(C)N1C C#CCC(C)(CC)C(=O)NC1CN(C(=O)CCS(C)=O)CC1CC(C)(C)C N1(C(COCCOCC#C)=O)CC(CNC(c2cncc(C)c2)=O)C2(CCC2)C1 c1(OCC)ccnc(NCC2CCN(C(=O)CCOC3CCOCC3)C2)n1 C1(N(C(C(COC)(C)C)=O)C)CC2CCC(C1)N2C(c1cncc(SC)c1)=O c1(C(=O)NC(CNC(C(C)C2CCCC2)=O)C2CC2)coc2c1C(=O)NCCC2 CC(C)(CC#N)C(=O)Nc1cccc(NC(C2CC3CCC2C3)=O)c1 c1(OCCC)ccc(NC(=O)Nc2ccc(-n3cncn3)cc2)c(C)c1 C(=O)(C#CC(C)(C)CNC(C1(C)CCCCO1)=O)NCCS(CC)=O c1(C(N2CC3C(NC(C(CC=CC)C)=O)(C3)C2)=O)ccc2nc(O)n(CC)c2c1 C(=O)(CCC(=O)NC(CC1CCOCC1)C(=O)N(CC(C)C#N)C)NCC N1(CCC)CCCC1C(=O)NC(C)(C)C(=O)NC1CCCC1CN(C)C C1(OC(C)=O)CCN(N2CCC(C)(F)CC2)CC1 CCCC(CCC)CC(=O)NCCC1CC(NC(c2cn(C(C)C)cn2)=O)C1 c1(C(=O)NCCC2(NC(C3C(CC)OCC3)=O)CCC2)ccc2oc(C)nc2c1 c1(-n2cc(CC3N(C(C)=O)CC(OCc4ccccc4)C3)nn2)nccc(Br)c1C C1(CNC(C2(OC)CC2)=O)CC(NC(c2ncccc2Cl)=O)C1(C)C N1(C(c2cn3ccccc3n2)C(=O)NC)CCc2[nH]nc(CO)c2C1 Cc1c(C(=O)NC2CC(NC(c3ccccc3)=O)CC2O)ccn1C C1(CNC(C(C)(C)C2CC2)=O)CN(C(=O)CCCN2CCCC2)C2(CCC2)C1 C1(OCC)CC2(C1)CC2C(=O)NC1CC(NC(c2ccnn2C(C)CC)=O)C1 CC1CN(C(c2ccnn2C)=O)C(C)CN1C(=O)CC1COCCO1 c1(C(N(C2CCC(NC(=O)CSC(F)F)C2)C)=O)conc1C1CC1 S(=O)(=O)(c1ccccc1)N(C(C(C)NC1CCCN(CCC#N)C1)=O)c1nccs1 c1(CC)ccc(C)cc1NC(=O)C=CCC1(NCC)CCC1.C1(C)(C=O)OCCO1 Nc1cc(C(=O)NCCC2(O)CN(C(C3CC3C(F)F)=O)C2)ccc1F N1(C(C=C(C)C(C)(C)C)=O)CC(C)(C)OCC1CNC(=O)C(F)=C1CCCC1 CC(O)C(C(=O)NCCN(C(=O)C(c1ccccc1Cl)C)C1CC1)N(C)C c1(C(=O)OC)cc(C)c(C(=O)NC2(CO)CCN(C(C3(C(C)C)COC3)=O)C2)o1 CC(C)(C)C(O)C(=O)NCC1COCCN1C(=O)Cn1cc(F)ccc1=O C(C(C(=O)Nn1cnn(CC)c1=O)CC(C)C)NC(C(OC)OC)=O c1(C(=O)NC2CCN(C(c3cccc(C(F)F)c3)=O)CC2)ccc(F)c(F)c1F C1(C(N2C(CNC(CC3(COC)CC3)=O)CC(C)CC2)=O)CCc2nc(C)sc2C1 Cn1cc(Br)c(C(=O)NCC2CCCC2NC(=O)Cn2nnc(=N)[nH]2)n1 CCC(CC(=O)N1CCCC1CNC(=O)Cc1ccc(Cl)cn1)c1ccccc1 N1(C(C2(C)CC=CC2)=O)CC(C(=O)NCCCS(N)(=O)=O)C2(CC2)C1 C1(C(N2CC(N(C(C3CN(CC(C)C)C3)=O)CC)C2)=O)CCC(N=[N+]=[N-])C1 c1(C(=O)NC2CN(C(CC=C)=O)CC2C2CC2)cc2c(Br)cccc2c(=O)o1 N1(Cc2ccc(C)nc2)CCCN(Cc2cnc(N(C)C)nc2)CC1 c1(C(=O)NCC(C)N(C(=O)C(F)C2CCOC2)C)ccc(C#N)cc1F c1(OC)cccc2ncnc(N3CCC(O)(C(C)NC(c4ccnn4C)=O)C3)c12 c1(OC)cc(CCC(=O)NCC2(F)CCC(CNC(=O)CC3CC3)C2)ccc1Cl C1(NC(CCOCCC)=O)CCC2(CCN(C(=O)CC(C)C)C2)C1 C1(C(=O)NCCCN(C)C(C2CCCC(=O)N2)=O)CC12CC(F)(F)C2 C1(C(CC(C)C)NCC(C(F)F)n2cccn2)CCCCCC1 c1(C(N2C(CN(C(=O)C=C(C)Cl)CC)CCCC2)=O)ccc2oncc2c1 C(CC)(CC)(CCNC(=O)C(C)(C)CC)NC(c1cccc(CC)n1)=O N1(Cc2ccc(OC)c(I)c2)CC(C(=O)NCC2CCOC2)CC(F)(F)C1 c1(N(C)C)cccc(C(=O)NCCCC2(NC(C3CCC3(C)C)=O)CC2)c1 CCCC(CCCO)C(=O)N1CCC(C)(NC(c2cccc(S(C)=O)c2)=O)C1 C(=O)(C(C(=O)N(CC(O)CNC(c1cncn1C(C)C)=O)C)OC)OC c1(C(N2CCCC(N(C(CC(COC)(C)C)=O)C)C2)=O)coc(S(N)(=O)=O)c1 C1(NC(C(C)CC2CCCC2)=O)C=CCC(C(=O)NCC(C)(O)CCO)C1 C(c1cnn(C)c1)=CC(=O)NC(C1(O)CN(C(C2CC2c2ccnn2C)=O)C1)C C(=O)(CC(C)CC(C)(C)C)N1CCN(C(c2ccnc(OC)n2)=O)C(CCO)C1 c1(OC)ccc(C(=O)NC2CCCC2NC(=O)COc2cccc(Br)c2)nn1 c1(C(N(C2CC(NC(=O)CO)C2)C)=O)cccc2c(Cl)c(Cl)sc12 C#CCC(C)(C(=O)NCC1COCC1(C)C)NC(c1ccon1)=O c1(CNC(C(C)(C)NC(c2n(CC)ncc2)=O)=O)cccc(Cl)c1 CCCC(C)(CC)NC(=O)C(c1cnn(C)c1)NC(=O)Cn1nccn1 N#Cc1c(F)ccc(F)c1NC(C1CC(CC2CC2)C1)=O c1(C(N2CC(NC(C(C)OCC3CC3)=O)C3(C2)CC3)=O)cn2cccc(Cl)c2n1 c1(NC(CC2(COC)CC2)=O)ccc2c(C)[nH]nc2c1 c1(COC)ccc(C(=O)NC2CCC2c2cn(C(C)C(=O)O)nn2)cc1 c1(CC)nc(C(=O)NCCC2(O)CN(C(=O)Cc3sccc3C)C2)co1 N1(C(C(CSC)C)=O)CC2CCCN(C(c3c(F)ccc(F)c3O)=O)C2C1 C1(CC)C(C(=O)NC(C)CS(C)(=O)=O)CCCN1C(c1ccc(CO)s1)=O C1(C(=O)NC(CN(C)C(c2ccc(C(C)(C)C)[nH]2)=O)(C)C)CCCOC1 N1(C(C2C(C)(Br)C2)=O)CCC(OCCNC(=O)CC2CC=CC2)CC1 C1(NC(=O)CC2C=CCC2)CN(C(=O)C2=CCOCC2)C2(CCCCCC2)C1 C1(C(=O)NC2CC(CC(N3CC(CC(=O)N(C)C)C3)=O)C2)CCCC1(C)C CCCC(CCC)=CC(=O)NCCC1(O)CN(C(=O)C(n2cc(Br)cn2)C)C1 c1(C(N2CCC(CC(C)NC(C(C(C)C)C)=O)CC2)=O)ncn2cccnc12 c1(C(=O)NC2C(NC(C3(CC=C)CCCC3)=O)C2)ccc(P(C)(C)=O)s1 c1(C(N2CC(CCNC(C(C=C=C)C)=O)C2)=O)cc(C)c2sccc2c1 Cc1cccn1C(=S)c1ccc2cc1N(CCNC(C)CC)C2=O Cc1cc(N2CCc3c(nnn3C)C2)nc(=NCC2(N(C)C)CCC(=O)N2)[nH]1 C1(C)(C(=O)NC2(CC=C)CN(C(=O)Cc3cc(Cl)cs3)C2)CC(C)OC(C)C1 C(=O)(C(C)P(C)(C)=O)N1CC(CN(C)C(c2cc(OC)cs2)=O)OCC1 c1(C(N2CC(OCC(=O)Nc3cccc(C(C)=O)c3)C2)=O)c2c(nn1C)CCC2 Cc1cc(C(C)CC2(c3ccsc3)CC2)cc(C)c1.C12CCN(CC1O)C2=O C(=O)(CC(C)(C)C#N)N(CCC(=O)NCC12CCCCC1C2)C(C)C Cc1ccc(F)cc1Cn1ccnc1-c1cccc(-c2ccncc2)n1 CC1CCCCC1NCCNC(c1ccccc1)=O N1(C(c2c(=N)[nH]cc3c2CCC3)=O)CCC2CN(C(C3C(Cl)(Cl)C34CC4)=O)CCC12 Cc1ccc(F)c(C(=O)N(CCNC(c2ccccc2N2CCCC2)=O)C2CC2)n1 N1(C(C2CC(C)C2)=O)CCC(OCC(N2CC(NC(=O)C(C)C)C2)=O)CC1 C=C(Cl)CCC(=O)NC1CC(N(C(=O)CC(C)C2CC2)C)C1 n1(CCC(=O)N(CC)CC)cc(C#CCNC(=O)C(F)n2cccn2)nn1 CCC(CC(=O)N1CCC(N(C(=O)C(C)(C)C(=O)OC)C)C1)CC(F)(F)F n1(CCC)cc(C(=O)NCC(F)CNC(c2cncc(C(C)C)c2)=O)c(C)n1 Cc1ccc(C(N2CC(NC(c3nc(Cl)sc3C)=O)C(C)C2)=O)cc1F O=C(C#CC1CCOC1)NC1CCC2CN(C(c3ccc(O)cn3)=O)CC12 C(=O)(C1CCCn2nccc21)NC(CC)CNC(=O)C(C)Cc1cnc[nH]1 N1(C(c2ccc(CCN3CCN(C)CC3)cc2)=O)C2C=CC(C2)C1CO C1(NC(c2cc3ncccc3s2)=O)CCC2CCN(C(c3nsnc3O)=O)C12 c1(C(N2CCCC(NC(C=C(C)C)=O)C2C)=O)cccc2c1CCC2 Cc1ccc(I)c(CNC(=O)CCc2cc(-c3ccccc3Br)no2)c1 c1(C(=O)NC(CC)CNC(=O)C(C)(C)C2CCCCO2)cccn2cnnc12 c1(C(=O)NCCN(C2CCCCC2)C(C2CCC(F)C2)=O)ncncc1Br CC1(CNC(c2cnn(CC(F)F)c2)=O)COCCN(C(=O)C=CC(F)(F)F)C1 c1(C(=O)NCC23CC2CN(C(=O)CC2CCCOC2)C3)cnc2c(F)cccn12 N1(C(C=C(CC)C)=O)CC2CCN(C(=O)C=CCOC)CC2C1 Cn1ncc2ccc(C(=O)NC3CCC(CNC(=O)C(F)(F)C(F)F)C3)cc12 NC12CCCC1CN(C(=O)C(N)CCc1cnc[nH]1)C2 Cc1cc(Br)c2oc(C(=O)NCCC3CN(C(C4(N(C)C)CC4)=O)C3)cc2c1 C1(C(=O)NCC(C=C)(C)C)CC(O)CN1C(=O)CNC(=O)CCC N1(C(c2cc(CC)no2)=O)CC=CCC1C(=O)NC(CC)C(C)(F)F c1(C(=O)NC(CC(C)C)(C)CNC(=O)C(C)S(C)(=O)=O)ccc2c(c1)CCCC2 c1(-c2cn(CCC3CC(NC(c4c(C)nccc4)=O)C3)nn2)ccc(Cl)cc1Cl CC(CCCCNC(=O)COCC1CCC1)NC(C1CC1(C)C(F)F)=O CCCC(C(=O)NCC(CNC(c1cncc(C(=O)OC)c1)=O)CO)N(C)C c1(C(N2C(C)CC(NC(C(CC=CC)C)=O)C2)=O)ccn2c(C)cnc2c1 C1(C(=O)NCCN(CCC)C(C)C)(CNC(c2ccc(N)cn2)=O)CCCCC1 Cc1nn(C)c(Cl)c1C(N1CC2C(CNC(=O)CC3CCC(C4CC4)O3)C2C1)=O C1(CNC(C(C=C)(F)F)=O)CN(C(=O)C(c2ccc(C)cc2)=O)CCC1(F)F C1(C(C)C)COCCN(C(=O)Nn2cc(CCN3CCOC3=O)nn2)C1 CON(CCC(=O)NC1CCCN(O)C1=O)C(=O)c1cnc(C)[nH]c1=N C1(NC(c2c(OC)ccc(C)c2)=O)CCC2CN(c3snc(C)c3C#N)CC2C1 CC(C)CCC(F)C(=O)N1CC(C)N(C(=O)CC(Cl)Cl)CC1C Cc1cc(=NC2CCCC(NC(c3cccnc3)=O)C2)c(C#N)c[nH]1 C1(CNC(CC=C=C)=O)CCN(C(c2cc(Cl)sc2Cl)=O)C(C)C1 C1(NC(c2cnc(C(F)(F)F)cn2)=O)CC(C)N(Cc2ncc(C(=O)OC)s2)C1 C12(C(N3C4C(CNC(=O)C5=CCSC5)C(CCC4)C3)=O)CCCCCC1OCC2 C(=O)(C(N=[N+]=[N-])C(C)C)N(C12CCC(CC1)C2)CCNC(c1c(C)ccnc1)=O N1(C(C(C=C)O)=O)C2CC=C(C(=O)Nc3cc(O)ccc3OC)C1CC2 C#Cc1cnc(C(N2CCC(CC)C2CNC(=O)C(C)NC=O)=O)c(C)c1 c1(C(CN2CCOC(CSn3c(C)csc3=O)C2)NC)cc2cc(Br)ccc2o1 C(=O)(CS(=O)(=O)CC(C)C)N1CCN(C(C(C)OCOC)=O)C(CC2CC2)C1 Cc1c(C(=O)NC2(C#N)CCN(Cc3ccc(F)c(F)c3)C2)ccc(F)c1F C(=O)(CCCS(N)(=O)=O)NC(C)CC1CN(C(c2ccc3c(c2)CC3)=O)C1 c1(C(=O)NCC(C2CCCC2)NC(C2C(CC)OCC2)=O)cc2n(n1)CCOC2 N1(C(C(CO)N(C)C)=O)CCC(F)(F)C(CNC(=O)Cn2cc([N+](=O)[O-])cn2)C1 C(C(CC1CC1)C(=O)NC1CCCC(C(C)C)C1)NC(C1CC(N(C)CC)C1)=O C1(C(=O)NCC(C)NC(N)=O)CCCC1c1cnn(C)c1.C1(=O)CCCN1 C(=O)(C(CC(C)(C)C)N1CCC(OCc2ccc(SC)cc2)C1)OC N1(C(C(C(=O)OC)(C)F)=O)CCN(C(=O)COCC(C)C)CC(C)C1 C1(C(=O)NC2C(C)CCN(C(=O)Cn3ncnn3)C2)=CN=C2C=CC(Cl)=CN2C1 CC1CC(NC(=O)CCN(C(C)=O)C2CC2)CO1.C1(N)COCC1SC C1(NC(C(C)SCC)=O)CN(C(C23CCOC2CCOC3)=O)Cc2nccn2C1 C(=O)(C(C(C)C)C(C)C)NC(CCNC(c1c(-c2cc(C)no2)ocn1)=O)C c1(N2C3CN(C(CCC=C)=O)CC2CC3)nc(O)c2c(ncn2C)n1 C(=O)(C(C)(C)CCCNC(=O)C(C)CC#N)N(CCOCC(C)C)C1CC1 c1(CN2CCCC(CC(=O)Nc3c(Cl)ccnc3Br)C2)ncc(F)cc1F c1(C(=O)NC2CC3(CC(CNC(C(C(C)C)O)=O)C3)C2)nccc2ncccc12 c1(C(N2CC(CCNC(C3(CC)CCCC3)=O)OCC2)=O)c(C)cc(=O)oc1C CCC(CC(=O)NCCNC(=O)Cc1csc(CSC)n1)C(F)F C1(C(=O)NC2CN(C(CS(=O)(=O)NCC)=O)CC2F)CCn2c(C)cnc2C1 c1(OC)ccc2[nH]cc(C(=O)NCC(O)CN(C)C(c3cnsn3)=O)c2c1 C1(NC(c2cc(C)cc(Cl)c2)=O)CC2CC1CN(C(C1CC(C)CCO1)=O)C2 N1(C(C(N2C(CCSC)CCC2)=O)=O)CCOC(NC(c2ncsc2C)=O)C1 N1(CCC(=O)N(CC(CNC(C=C(C)C(C)C)=O)O)C)CCN(C)CC1 C(=O)(C(CCc1ccccc1)C(C)(C)C)C1C2(CC(C(=O)OC)C2)C1 c1(SC(C)C)ccccc1CNC(N1CCN(C2CCS(=O)(=O)C2)CC1)=O Cn1ncc2c1CCC(C(=O)NC1(C)CCCN(C(C3(C4CCC4)CC3)=O)C1)C2 N(S(=O)(=O)N(C)C)CC(=O)NC(CC)CNC(C1CC1CCOC)=O C(C)(CC(=O)NCC12CC(NC(=O)CCCn3ccnn3)(C1)C2)SC Cc1ncc2n1CC(C(N1CCC(N3CCN(C(=O)C(C)CF)CC3)C1)=O)CC2 c1(OCC)cnc(C(N2CCCC2CN(C(=O)CC2CS(=O)(=O)C2)C)=O)cn1 C1(CNC(=O)CCC2CCCCC2)CN(C(=O)C(O)CC2CCOCC2)CCO1 Cc1cccc(C2(O)CCN(C(=O)OC(C)(C)C)C2)c1C.C12CC(C1)NC2 c1(CC(=O)NC2CCCN(C(C(C)OCC)=O)C2C)c[nH]c2c(C)cccc12 Cc1nn(C)c(C)c1C(C)C(=O)NC1(C)CN(CCCC2CCCC2)CCO1 C1(CC)CN(C(=O)CC2CC2CNC(C2COC(=O)N2C)=O)CCS1 c1(CC)nc(C)c(NC(=O)COCCCOCc2ccccc2)cc1C c1(N(Cc2cc(C)on2)CC2CCCO2)cnc(C(C)(C)C)nc1 c1(C(=O)NCC(C(=O)NC2C(OCC)C(O)C2)CC2CC2)ccc(C)c(F)c1 c1(OCCOC(Cn2nc(C)c(Cl)c2)=O)nc2cc(Cl)ccc2s1 C1(CNC(c2cn(C)nn2)=O)CCC(NC(C2(CC3CC3)CCCO2)=O)CC1 c1(CO)ccccc1Cn1cc(C2CCCN2C(=O)C(Br)Br)nn1 c1(C(=O)NCC2CCN(C(C3CCCCC3)=O)CC2)ccc2c(c1)CCNC2=O C(C(COC)C(=O)NCC1COCCN1C(c1cccc(=O)o1)=O)OC c1(OC)nc(C(=O)N(CC(O)CN(C)C(C2CC2Cc2ccccc2)=O)C)ns1 Cc1cc(Br)cc(CNCC23CC2CN(C(c2cccnc2I)=O)C3)n1 Cc1ccc(N)cc1S(=O)(=O)NC1C2CCC(C2)C1C(=O)O C12(C(=O)NCC3C(C)CCN3C(=O)CN3CCCCCC3)CCC(F)(CC1)CC2 C(C)(CC(C)N=c1[nH]cnc2cc(Br)sc12)NC(C(C(CC)C)O)=O c1(CC(=O)NCc2cn(C(C(=O)OC)C)nn2)ccc(F)nc1 CCC(CC)(CC)C(=O)N(CCCC(=O)NC(c1ccco1)CO)C C(C)(C)(CCCC(=O)NCc1ncc(F)cc1F)NC(C1CN(C)C1)=O c1(NC(c2cc(OC)ns2)C)cc(N2CCOCC2)nc(C)n1 N1(C(c2c(C)nsc2)=O)CCC(C2CCN(C(c3cc(N)ccc3Cl)=O)CC2)C1 c1(C(=O)NCC2N(C(CCNC(=O)OC)=O)CCC2C)cc(C)nc(C)n1 C(=O)(C(C)C(O)C(C)C)N.c12nc(cs1)C(=O)NC1CC(C1)NC2=O.C=CCOCC C(=O)(CCCC(=O)N(C)C)NC1(C(=O)NC)CSC1.C12CCCCC1NC2=O c1(C(N2CCC(NC(c3cccnc3O)=O)C2)=O)cncc(OC2CC2)c1 N1(C(C(c2ccc(Br)cc2)=O)=O)CCSc2ncccc21.N12CC(C1)C2=O C1(NC(C(=O)NCc2ccccc2Cl)=O)CC(O)CN(C(C2CCCCC2)=O)C1 N1(C(c2cnc(C(C)C)[nH]2)=O)C2CCCC1CN(C(=O)C(C)(C)C(C)(F)F)CC2 N1(CC)CCC1C(=O)NCCN(C(=O)C(C)N(C)C(C)=O)Cc1ccco1 C(C(=O)NCCC(C)CCNC(c1ccns1)=O)(C(C)C)NC(=O)OCC Cc1nscc1CNC(C1(N(C)C(C2CCCCS2)=O)CC1)=O C1(CCC(=O)NCC(=C2CN(C(C(C)OC3CCCC3)=O)C2)F)CCC(=O)N1 c1(OCCC(=O)N(CCNC(C(C=CCCC)O)=O)C)ccccc1O c1(C(=O)NCC=CCNC(C(C)OCC)=O)c(C)cc(OC)cc1F c1(NS(C)(=O)=O)ccc(C(=O)NC2(CF)CN(C(c3cc(F)n(C)n3)=O)C2)cc1 N1(CC(C)(O)C(F)(F)F)CCC2(C)C(C1)C2(Cl)Cl c1(NC(C2N(Cc3ccn(C)n3)CCSC2)=O)ccc2cnoc2c1 c1(CSC)cc(C(=O)NCC2CN(C(=O)C=C(C)Cl)CCCO2)ccc1F N1(C(CSC)=O)CC2CC(N=c3nc(C4CCOCC4)[nH]s3)CC1C2 Cc1cnc(N2CCC(NC(C3(C(F)F)CCC3)=O)CC2)nc1O C1(NC(C2(C(CC)=O)CC2)=O)CCN(C(C2CC3CC(OC)C3C2)=O)C(C)C1 CN1CCCC1(C)C(N1CCCC1C(C)(C)CNC(c1ncc(Br)cn1)=O)=O C12(CCNC(CC3(NC(C)=O)CC3)=O)CCC1CN(C(=O)CCC(C)O)C2 c1(NC(C2CN(C(C3CCCO3)=O)CCC2O)=O)cccc2cccnc12 Cc1cccc(CCNC(=O)C(CCN(C)C)NC(C2CCCC2O)=O)n1 c1(CC(C)C(=O)NC2(C3CN(C(=O)CC(C)(F)F)C3)CC2)ccc2c(c1)CCC2 c1(C(C)NC(C2CCCN(c3cc(O)ncn3)CC2)=O)cccc([N+](=O)[O-])c1 C1(OC2CN(C(C3(C)CC3)=O)C2)CCN(C(c2nocc2Cl)=O)CC1 CCC(CN(C)C)C(=O)NC(c1cc(C(=O)NC(c2ncc(F)cn2)C)on1)C N1(C(C(C)OC)=O)CCOC2(CCN(c3ncnc4c3ncn4CCO)C2)C1 n1(CCC)ccc(C(=O)NC2CCC(NC(c3cc(Br)no3)=O)C2)n1 CC(C)CC(C)CC(=O)NC1CCCC1C(=O)NCCn1cncn1 N1(C(C2(O)CCCC(C)CC2)=O)CC2(CCC(NC(C3COC(=O)N3)=O)CC2)C1 c1(C(CN(CC(=O)NC(c2cccc(C)c2)N(C)C)C)C)ccc(F)c(Br)c1 c1(CNC2CCC(C(N(CC#N)CC#N)=O)CC2)cc(Br)cc(F)c1F N(C1CCOc2ccc(Br)cc21)C(C1CCC(CNC(c2c(C)ncs2)=O)CC1)=O C1(CO)CCCN1C(=O)C=CCOCC.C12CC1C(=O)N(CC)C2 Cc1nc2cc(C(N3CCN(C(C4CC(O)C4)=O)C(CO)C3)=O)cnc2s1 c1(-n2cc(CNCCCC3CCN(S(C)(=O)=O)C3)nn2)cccc(F)c1 c1(C(N2C(C(=O)NC3CC(C)OC3=O)CCC2)=O)cc2ccccc2o1 C1(C(=O)OCC(=O)NC(C=C)CC)CCOCC1(C)C CC#CCCCC(=O)NCC1CCN(C(=O)CC2CC=CCN2C)CC1O c1(C(=O)NCC(n2cc(C(CO)CC(C)(C)C)nn2)C)coc2cccc(O)c12 CC(C)(C)CC(O)C(=O)NCCN(C(c1nc(Br)c[nH]1)=O)C1CC1 c1(C(=O)NCCN(C(=O)COC2CCCCC2)C)ncc(Cl)cc1Cl c1(CN(C=O)Cc2ccccc2)ccc2c(c1)CC2.C1(OC)(OC)CCC1 c1(C(=O)NC2C(C)CCN(C(C3(n4cccn4)CC3)=O)C2)nc2ccccc2s1 C1(C(=O)Nc2cccc(C(C)=O)c2)(OC)CCN(CCCC(N)=O)CC1 N1(C(COC2CN(C(C(C)OCCOC)=O)C2)=O)CCOC(C(C)(C)C)C1 Cn1c(=N)[nH]c2cc(C(=O)NC3CC3NC(=O)C(F)=C3CCCC3)ccc12 N1(C(C=C2CCC(C)C2)=O)C2CCC1CN(C(=O)CNS(=O)(=O)C1CC1)C2 C(C(=O)OCc1ccccc1)(C(=O)O)NC1C(CC)C1 c1(C2C(C(N3CCCC(N(C)C(c4cocn4)=O)C3)=O)C2)ccc([N+](=O)[O-])cc1 c1(C(N2CCOCC(NC(c3c(C)onc3)=O)C2)=O)nc2cncnc2[nH]c1=O N1(C(c2cccc(OCC)c2)=O)CCN(C(C2(F)CC2)=O)C2CCCCC12 N1(C(C2(C)CCC2)=O)C(C(N2CCC(O)C(C)(O)C2)=O)C2CC(O)C1C2 C1(CNC(C(C)(C)C2CCN(C(C3CC=CCO3)=O)C2)=O)CCC(O)CC1 N1(C(c2nccc(C)c2)=O)CC(NC(=O)CN2CCOCC2)CC(F)(F)C1 N12CCN(CC1)C(=O)CN1CC2C1.C12(NS(=O)(=O)C3CC3)CCCCC1C2 C(=O)(C(C)CC(F)F)NC1C(OC)CN(C(c2ccnn2C)=O)C1 N1(C(Cc2c(CC)n[nH]c2CC)=O)CCCC(N=c2nc(C)nc3[nH][nH]cc2-3)CC1 c1(C(=O)NCC(CNC(c2c(CC)occ2C)=O)F)ccc(=O)n(C2CC2)c1 N1(C(=O)C2CC2)CCN(C2(CC(N3CCC(c4ncco4)C3)=O)CCC2)CC1 C1(C(N2CC(C(C)NC(C3CC(=O)N(O)C3)=O)C2)=O)CN(C)CCN(C)C1 c1(CC)cc(C(=O)N(C2(C(=O)NC3CC(n4ccnn4)C3)CCC2)C2CC2)no1 c1(CSCC)ccc(OCC(N2CC(SC3CCOC3=O)C2)=O)cc1 c1(NCCNC(C(CC)N(C)C(c2cc(CO)on2)=O)=O)ccccc1C c1(C(=O)NCC(CC)NC(=O)C(O)C2CCC2)cc(COC)[nH]n1 C=C1CC2CCC(C1)N2C(=O)C(CNC(C1(c2ccno2)CC1)=O)CC c1(C(C(=O)NC2CCOCC2)N(C2(COC)CC2)C)cccc(SC)c1F N1(C(Cc2c(C)ocn2)=O)CCC(C2CN(C(c3coc(O)n3)=O)C2)CC1 CCCCS(=O)(=O)CC(=O)NCC1CC2CCC(C1)N2C(=O)C=CC1CCCO1 Cc1ccc(C2(NC(C3CC3c3ccc(Br)o3)=O)CC2)cn1.c12cn(C)nc1OC2 c1(C(=O)NCCC(C)OC)ccc2c(n1)CCC(C)C2 C#CC(C(C)OC)NC(c1coc(CNC(C2(SC)CC2)=O)n1)=O C1(C(=O)NCC2CCCC2NC(=O)CCNC(=O)CO)(OC)CCC(C)(C)CC1 N1(C(c2cc(C)c(C)o2)=O)CCC(NC(c2cnc(Cl)c(N)c2)=O)C(CO)C1 C(=O)(CS(=O)(=O)CC1CCCO1)N(C1CCCC(NC(C)=O)C1)C C(=O)(CC(C)C(F)(F)F)NC1CCCN(C(c2n(C=C)ncc2)=O)CC1 c1(C(N(CC=CC(=O)N(C(C#C)C2CCC2)C)C)=O)ccc([N+](=O)[O-])o1 CC1=C(C(=O)NCC2CCN(C(=O)Cc3cnn(C)c3)C23CCC3)CCS1(=O)=O c1(C(N2CC(N(C(=O)C=C3CCOCC3)C)C(O)C2)=O)ccc(F)cc1C#N c1(C(=O)NC(CNC(C2C(COC)(COC)C2)=O)(C)C2CC2)ncn(C)c1C c1(CC(=O)NCC(C2CC2)NC(CCc2cc(C)on2)=O)ccc2nsnc2c1 C12(NC(CCCOC)=O)CCC(NC(=O)C(c3cccc(F)c3)C)(CC1)C2 c1(C(N2CC(C3(NC(c4ccc(C)cn4)=O)CC3)C2)=O)cc(Cl)cc2c1OCC2 C1(NC(C(C)CC(N)=O)=O)CC2(CCC(NC(C3CCCCN3N=O)=O)CC2)C1 Cc1c(C(=O)NC2CC(C)CN(C(=O)C(C)C)C2)cc(-c2ccccc2)n1C N1(C(c2ccc(OC)cc2F)=O)CCCC2(CCCN2C(c2cc(C)ns2)=O)C1 CCC(C)CC(C)C(=O)NCC1CC2(CC(NC(=O)CNS(=O)(=O)N(C)C)C2)C1 N1(C(C(c2ccccc2)C)=O)CCC2(CC1)CN(C(=O)CC(C)F)CC2CO N1(Cc2cc(OC)no2)CCCC2(CC1)CNC(=O)C2 c1(C(N2CC(C)(NC(c3cc(C)sn3)=O)C2)=O)cc2c(C)c(Cl)ccc2[nH]1 C1(C(=O)NCCC(C)NC(c2c(O)cccc2Cl)=O)CCCCC1C1CC1 N1(C(CC(CNC(CC2C(C)OCC2)=O)(C)C)=O)CC2CCCC(O)C2C1 C(=O)(N=c1cc(C)n(C2CC2)[nH]1)c1c(C)cccn1.c12ocnc1CNC2 C1(C(N2CCC(C)(NC(=O)CCc3cn[nH]c3)C2)=O)CC(C2CCC2)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CC2CC2(CNC(=O)Cn2ccnn2)C1 Cc1ccc(O)c(CNC2CC(NC(c3cnc(CO)s3)=O)C2)c1 N1(C(C=CC(C)(C)C)=O)CC2(CC(CNC(C3C4CCC(=O)C34)=O)C2)C1 CCC(CCN=c1[nH]c2c(c(=NC3CCC(OC)CC3)[nH]1)CC(C)CC2)OC c1(C(=O)NCCCN(C(C2CC2O)=O)CC)ccnc2c1CCC2.c1(SC)ccccc1 C(=O)(CP1(=O)OCC=C1C(=O)CCC(c1nc2ccccc2s1)(C)C)NCC CCC(CO)(C(=O)NCc1ccc(C(C)NC(C2CCCC2C)=O)cc1)OC C(=O)(C1CCC(=O)c2ccccc21)NCCOCCCNC(c1ncc(C)s1)=O N1(C(=O)NC2CCN(C(CCC)C)CC2)CCn2cccc2C1C(=O)OCC c1(CC(=O)NC(C)C=CC(=O)N(C)C(c2ccccn2)C)cnnn1C c1(C(N2CC(OCCOCCOC)C2)=O)cccc(-c2ccc(O)nc2)c1 C(=O)(C(O)CN1CCOCC1)NC1CN(C(C2C(C)C2C)=O)C1 C1(S(C)(=O)=O)(C(N(c2ccccc2)C)=O)CNC1.C12CCC(CC1)N2 c1(C(=O)NC(C)CCN(C)C(c2cc(CO)[nH]n2)=O)cc(C2CC2)ccc1Cl c1(CNC2(c3n(Cc4nnn(C)n4)nnn3)CC(C(F)F)C2)ccc(Cl)c(Br)c1 c1(C(=O)NCc2c(C(N(CC(C)O)CC)=O)occ2)cc(N)cc(F)c1 C1(C2CCN(C(C3CN(C)CC3C)=O)CC2)(NC(CCC(=C)Cl)=O)CCC1 C1(CNC(CCOCC#C)=O)CC2(CC2)CN1C(=O)C(C)C(=O)OC(C)(C)C C(=O)(C(CNC(c1ccc[n+]([O-])c1)=O)CCC)NC(CCC)CC C(=O)(CC(C)(C)C=C)N1CCC(CC#C)(C(=O)NCCCCC2CC2)C1 N1(C(C(C)OCCOCC)=O)CCCCC(N(C(=O)C2=COCC2)C)C1 C(=O)(C(C)S(N)(=O)=O)NCC1CCC(NC(CN2CCC(C(C)C)CC2)=O)CC1 Cc1ccc(S(=O)(=O)CCC(=O)N2CCC(C)(NC(C3CCCN3C)=O)C2)cc1 c1(NC)cc(Cl)ccc1C(N1CCCCC(NC(=O)CC(=O)OCCC(C)C)C1)=O C1(c2n(CCOC)nnn2)(NC2CSC2)CSCCSC1 c1(NC(C2N(C(C(C=C=C)C)=O)CC2C)=O)cc(F)ccc1O CCC(C(=O)NC(C(=O)NC(C)CC(F)(F)F)c1cccs1)C(C)(C)CC CCC(C)(C)C(C)CC(=O)N(C(CNC(=O)Cc1cccc(F)c1O)C1CC1)C C(=O)(CS(=O)(=O)C1CCCC1)N(CCCNC(C(c1n(C)ccc1)=O)=O)CCO c1(C(C)N(C(=O)C(=O)NC2CC(n3ccnn3)C2)C)ccc(Br)cc1 C12(C(=O)NCCc3cccc(O)n3)CCCC1CN(C(=O)CCc1nncs1)C2 N1(C(C2CC23CCC3)C(=O)NCC=C)CCCC(O)(C2CC2)C1 C1(C(=O)NC2CN(c3c(C)cncn3)CC2C)CCc2ccccc2C1 C12(CN3CC(O)C3)CCCN(C1)NC2.n12cc(nn1)C2 c1(NC)nc(C)ccc1C(N1CC(F)(CNC(=O)C(c2cn(C)nc2C)C)C1)=O C1(NC(=O)CCOc2ccc(F)cc2)CC2CN(C(=O)CCc3cscn3)CC12 c1(CCC)cc(C(=O)NC2CC(O)(CNC(c3occc3C)=O)C2)n[nH]1 c1(CN(C(=O)C(c2cncn2C)O)CCNC(C(CC)OC)=O)ccccc1C c1(CC)c[nH]c(C(=O)NC(CNC(C2CC2c2cccs2)=O)C(C)C)c1 n1(CC(=O)NC(C2CN(C(C(CC)NC(C)=O)=O)C2)C)c(C)cc(O)cc1=O C1(C(=O)NCC=C2CCN(C(=O)CCc3ccsc3Cl)CC2)CC2C=CC1CC2 C1(CC(=O)NCC(C2CCC2)NC(c2c(C)nn(C)c2)=O)CCCC2(CC2)C1 c1(C(=O)NCC2(C(C)NC(C=CC)=O)CC2)c(CO)n[nH]c1C C1(C(=O)NCCCC2C(C)C2)CCCCC1NC(=O)C(O)CN(C)C N1(C(CN(C)CC)=O)CC2CCCC2(NC(c2cc(SC)c(C)o2)=O)C1 c1(NC(=O)NC2C3(CC3)C23CC3)cc(Cl)nc(C2CCOCC2)n1 c1(C(C(=O)NCC(C)NC(c2ccc(N(C)C)cc2)=O)(C)C)ccc(F)cc1Cl CC1(NC(=O)CNc2ccccc2)CCN(C(C23CSC(C2)C3)=O)CC1 n1(CC)cc(NC(=O)COC2CN(C(=O)CC3CCC4CC34)C2)c(C)n1 c1(N(C)C(=O)NCC2CC(C(F)(F)F)CN2CCN)ccccc1N(C)C C1(C(=O)NCc2n(CC)ncn2)CC(F)CN1C(=O)C(C)c1ccco1 C(=O)(C(Cc1ccccc1)S(C)(=O)=O)N1C(CNC(C=NOC)=O)CCCC1 CC1(C(=O)NCC2CCN2C(C2CC(c3ccncc3)C2)=O)CCCC1(F)F N1(CC)CCCC(C(=O)NC2CC(NC(=O)Cc3ccc(C)cc3)C2)C1 Cc1c(Cl)cnn1CC(=O)NC1CC(F)(CNC(=O)CCOC2CCCCC2)C1 c1(CNC(=NC)NCC(O)(COC)COC)c(N2CCOCC2)ncnc1Cl c1(C(N(C2CCC(NC(=O)CCC(C)(C)C)C2)C)=O)ccc2nccn2c1 N1(C(CS(CCC)(=O)=O)=O)CC2CN(C(C34CC3CNC4=O)=O)CC(C1)O2 c1(C(=O)NC2CC(C)N(C(=O)C(=C3CCCCC3)F)C2)n[nH]c2ccc(F)cc12 c1(OC)cc(C(N2CCOC(CNC(c3cc[nH]c3)=O)C2)=O)cc(F)n1 C12(C(N(C3CCCCCC3)CCNC(C=CSC)=O)=O)CCC(CF)(CC1)CC2 CC(C)(CNC(C1CC2(CC2)CO1)=O)CCNC(=O)CCOC1CCOC1 N1(C(c2c(C)non2)=O)C(C(=O)NCCc2ncccc2C)CCC1C1CC1 C1(C(C)=O)CC(C(=O)NCCCCn2cc(-c3cnnn3C)nn2)C1(C)C c1(OC)ccnc(C(=O)NC2CCCC(NC(=O)C=C3CCC3)C2)c1N C1(C(N2CCC(C)(CNC(c3ccnnc3)=O)C2)=O)CC2(C1)OCCO2 N1(C(CCOCC#C)=O)CCN(C(c2cc(C)nn2CC)=O)CC1CC(F)(F)F C1(NC(CNC(=O)NC)=O)C(C)CN(C(C2(CC3CCC3)CC2)=O)CC1C C1(NC(C(C)c2cncs2)=O)CCN(C(=O)COc2cccc(F)c2)C1C c1(C(=O)NCC(C)N(C(c2n(CC)nnc2C)=O)C)c(F)c(N)cc(Cl)c1F C1(C(N2C(C)CC(CO)C2)=O)C2CC(O)C(C2)N1C(=O)CC1CCCC(=O)C1 c1(CSC(C)C(=O)NCC(F)CNC(=O)C=CCN2CCCC2)ccccn1 C(=O)(C1=CC2(CCOC2)C1)NC1(C)CC(NC(c2n[nH]c3c2CCC3)=O)C1 C1(CNC(c2scc(C)c2)=O)CC2(CCC2)CN1C(c1ccn(CCF)n1)=O c1(CC(=O)NC(CN(C(=O)CSC2CCCO2)C)(C)C)cc2cc(Cl)ccc2[nH]1 C1(C2CNC2)(NC(=O)C(Cc2ccccc2)Cc2ccccc2)CCC1 Cc1cc(C#N)cc(C(=O)N(CC(O)CNC(c2nc(C(F)(F)F)cs2)=O)C)n1 N1(C(c2csc(Cl)c2Cl)=O)CCN(C(c2cc(Cc3ccccc3)[nH]n2)=O)CC1 c1(C(=O)Nc2cc(C(=O)NCC(C)CN(C)C3CC3)[nH]c2)ncnc2cc[nH]c12 O=C1CC(CC(=O)NC2(C(F)(F)F)CC3(CCC3)C2)c2ccccc2N1 N1(C(C(C=C)OC)=O)CC2CN(C(=O)C=CSC)CCC12 C=CCC(Cc1ccccc1)C(=O)NCC(C)CN(C)C(c1cccc(C)n1)=O N1(C(c2cc3nc(C)sc3[nH]2)=O)CCN(C(=O)CN2CCCCC2)C2(CCC2)C1 C1(NC(C(c2cnccn2)C)=O)CCCN(C(c2c(Cl)csc2Cl)=O)CC1 C1(NC(C=COCC)=O)CN(C(C2CCCCC2O)=O)CC1Cc1ccccc1 c1(C2CN(C(C(C)N(C(C3N(CC)CC3)=O)C)=O)C2)nc(=O)o[nH]1 C1(NC(c2ccc(CNC(CC(C)CN(C)C)=O)cn2)=O)CCCC(O)C1O CC1OCCC1(C)NC(C1(CNC(=O)CNc2ncccn2)CC(C)(C)C1)=O CCC(CCC(=O)Nc1cccc(Cl)c1O)NC(=O)C(C)(C)n1cnnn1 C=CC(C)C(C)C(=O)NCC1(O)CCN(C(c2cn(C)nc2O)=O)CC1 CC(C)C(CNC(C1(NC(=O)Cc2cc(Cl)n(C)n2)CCCC1)=O)CO N1(c2n(CC(=O)NC)nnn2)CCOCC2(C1)CC2(F)F N1(C(Cc2ccc(C)cc2)=O)CCc2sc(-c3cnn(C)c3C)cc2C1 CCC(CCOC)C(=O)N1CCCCC1CNC(=O)CC1CC=CCC1 c1(CNC(=O)C(=O)Nc2cccc(C(F)(F)F)n2)cc(F)ccc1F c1(CNC(C2C(C(=O)N(CC#C)C3CC3)C2)=O)ccc(Br)c(Cl)c1 CC(C)C(C)(O)C(=O)NCC1CCN(C(=O)Cn2ncc(Cl)c2C)CC1O C(=O)(C(CC(=C)C)NC(=O)C(C)CC#N)NCCC(C=C)(C)C CCC(C)(C(=O)N1CCC(CC(=O)NC)C1)NC(=O)CCc1cncnc1C C(=O)(C1CCc2nccn21)NCC1CN(C(c2ccc(=NC)[nH]c2)=O)CC12CC2 C(=O)(CCCCCC(C)C)N1CC(CC)N(C(=O)CC2CC2)CC1 c1(NC(CC)CC(F)(F)F)[nH]c(=NC2CCCN(C)CC2)nc2ncn(C)c12 CCC(C)(C)C(O)C(=O)N(C1CCCC1C)CCSC1CC(=O)N(C(C)C)C1 C1(NC(c2ncncc2Cl)=O)(CO)CCCN(C(c2ccc(F)o2)=O)C1 c1(N(CC)CC)ccc(C(=O)NC2(C)CC(NC(=O)CC3C=CCC3)C2)cn1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC(C)(NC(c2[nH]nnc2C2CC2)=O)C1 N1(C(c2c(C)csn2)=O)CCC(CO)(CNC(C2CC2(C)C(F)F)=O)C1 CC1(C)CC(NC(C2C3CCCC23)=O)CN(C(C2CCCCC(=O)C2)=O)C1 C(C(C(C)C(C)C)NC(c1cnn(C(F)F)c1)=O)NC(c1ccc(C(C)=O)[nH]1)=O N1(C(C=C(C)C)=O)C2CCC(C2)C1C(N1CCOCC1C(C)(C)C)=O C1(NC(C(C(C)NC(c2ccc(C(F)F)o2)=O)(C)C)=O)CCOC12CCCC2 N12CC(CC(F)C1)C2=O.c1(C(=O)O)cccc(CNc2cnns2)c1 CCC(CNC(C1C2CN(C(c3ccccc3OCC)C)CC12)=O)CC(=O)NC c1(NCc2ncn(C)n2)nc2ccccc2nc1NCCC1(C)CC1 c1(NC2CC3CN(C(CC(=O)N(C)C)=O)CC32)ncnc2c(Br)cccc12 c1(NC(C2CC2C(=O)NC(c2ccc(Cl)cc2)CO)=O)cnn2cccnc12 C1(C2CC2)(N)CCN(C(=O)Cn2cccn2)C1.c1(NC(COCC)=O)ccc(Cl)cc1 N1(C(C(c2ccccc2)C)=O)CCCCCC1CC(=O)NCC1(N(C)C)CC1 c1(OCCN(C)C)ccc(C(N2CCC(C)(NC(=O)CNS(C)(=O)=O)C2)=O)cn1 CC1Cc2cccc(C(=O)NC(CO)C3(C)CC3)c2C1 C(=O)(C(C(C)(C)C)OCCOC)N1CC(C(NOCC(=C)C)=O)(CC=C)C1 c1(C(C)C)ccc(O)c(C(=O)NC2CCNC2CO)c1 c1(C(N(C2CN(C(c3nc(C)nn3C)=O)CC2O)C)=O)nn(C)c2ccccc12 N1(C(C2(COC)CCC2)=O)CC2(CCCC2NC(c2c(C)coc2C)=O)C1 N1(C(C2C(CC)CN(C(c3cnccc3C)=O)C2)=O)CCCC(CO)CC1 Cc1c[nH]cc1C(=O)NCC=CCNC(C1COC(C)C1)=O Cc1c(N(C(=O)C(O)CNC(C2(F)CC2)=O)C)cccc1F C1(NC(C2(O)CC(C)(C)C2)=O)CCCCCN(C(=O)CN2CCP(C)(=O)CC2)C1 N1(C(C(C=CCCC)O)=O)CC2(C)CN(C(=O)Cn3nnc(C4CC4)n3)CC2(C)C1 c1(C(=O)NCC(F)F)cc2ccc(-c3cc(O)c(F)cc3F)nc2[nH]1 C1(C(=O)NCCN(CCOC)C)CC(O)CN1C(=O)CNS(=O)(=O)N(C)C C1(CC(C)(C)CNC(=O)OC(C)(C)C)CCn2c(cnc2-c2ccccc2)C1 c1(N(CC(CC(C)C)NC(=O)CSC(F)(F)F)C2CC2)cc(=O)n(C)c(=O)n1C Cc1cccnc1CCC(=O)NCC1C(C)CCN1C(c1ccc(CF)cc1)=O CC(CC=Cc1ccccc1)C(=O)NCCNC(c1nscc1Br)=O c1(SCC(=O)N(CCC(C)NC(C(C)SC(F)(F)F)=O)C)nnnn1C1CC1 C12(C(=O)NCC3C(CNC(c4ccnc(C)n4)=O)C3(F)F)CCOC(C)(C1)C2 c1(C(=O)O)ccc2ccnc(Nc3c(F)ccc(-c4ccc(F)cc4)c3F)c2c1 C1(CC(=O)NC2CC2C2CCC2)CCN(C(=O)C=CC2CCOC2)CC1 c1(C(=O)NCC2CC(SC)C2)cc(CNC(c2ccns2)=O)nn1C c1(C(C)C)nc(C2C(OC(C)(C)C)C2)no1.C1(C(=O)OO)N(C=O)CC12CC2 c1(C(=O)NC2CC(NC(c3ccc(C#N)s3)=O)C2)cc2c(nn1)CCOC2 N1(C(CCc2cnc(C)o2)=O)CC12CCN(C(c1cccc(C(N)=O)n1)=O)C2 CC1(C(=O)NC2CCC(NC(=O)C=C3CC3)CC2)CCCOC1 N1(C(c2cc(C)[nH]c2C)=O)CC2CCCC1CN(C(C1CCCCC1)=O)C2 C(C(C)(O)CN(C)C)N(C(C)C(=O)OC(c1cccs1)=O)C(c1ccco1)=O.CO O=S(=O)(c1ccc(NC2CN(S(C)(=O)=O)C2)c(F)c1)N1CC2C3C=CC(C3)C2C1 c1(C(c2n(CC(=C)C)nnn2)NCc2csc(C(C)C)n2)nnc2n1CCS2 Cc1nc[nH]c1CC(=O)NCC(F)CNC(=O)C(C)CN(C)C C(CC(C)C(F)(F)F)NC(C(CCOC)NC(c1ncc(CC)cn1)=O)=O c1(C(=O)NCCCCCNC(c2c(C)cnnc2)=O)cncc2cnccc12 C1(CC=C)(NC(c2nocc2Cl)=O)CCN(C(=O)C(C)=CCO)C1 C1(NC(c2c(COC)noc2)=O)CCCN(C(c2ccc(O)c(Br)c2)=O)CC1 C(CN=C(NCC)NC1CCN(c2ccccc2)C1)N(C1C(OC)(OC)CC1)C Cc1ccccc1CCC(=O)NC1CC(C)(NC(=O)CCOC(F)(F)F)C1 CC(C)CC(CNC(=O)CC1(O)CCCCC1)C(=O)NCC1CC1C C1(C(N2C(C)CC(NC(c3cnns3)=O)C2)=O)Cc2ccccc2CO1 c1(C(=O)NC2CCC(NC(c3cn(C)nc3)=O)CC2)ccc2cccnc2c1O C1(CCC(N2C(C(C)C)CCC2)=O)CCN(C(C2(C)CCCCO2)=O)CC1 C1(n2cc(C(CCC)=O)nn2)CCCCC1N(C(=O)CCC1CCC(=O)C1)CC N1(C(CNC(C2C(C)C2)=O)=O)CC(C)(C)OCC1CNC(=O)CN1CC(=O)NC1=O c1(C(=O)NC2CC3(C(NC(C(CCC)OC)=O)C3)C2)cc2c(Cl)ccnc2s1 CN1CCN(C(C2C3CN(C(C4CC5(CCO4)CC5)=O)CC23)=O)C2CC12 N1(C(c2c(C)n(C)cc2)=O)CCN(C(C2CCCSC2)=O)C(C)C1 c1(OC)cccc(C(CF)N(CC(=O)NC(=O)NC(C)C)CCO)c1 N(C(=NCCCCCCC(F)(F)F)NC1CCCCC1)OC1(COCC)CCC1 Cc1scnc1CNC(=O)CNC(C1CC1(Cl)Cl)=O Cc1nc2c(-c3nc(-c4ccoc4)nn3-c3cnn(C)c3)ccnc2[nH]1 C12(CC(N3CC(N4CCN(C(CN5CC(C)C5)=O)CC4)C3)=O)CCCN1CCC2 c1(OC)ccc2oc(C(N3CC(NC(=O)C(F)C(C)C)C(F)C3)=O)cc(=O)c2c1 c1(OCC(=O)N(CCN(C(=O)Cc2n[nH]c(O)n2)CC)CC)ccc(Cl)c(F)c1 C1(CNC(=O)CC2CCCC2(F)F)CN(C(C2CCCC3(CC3)C2)=O)CCCO1 C#Cc1ccc(C(=O)NCC(O)CN(C(=O)CCc2nnc(S)n2C)C)o1 N1(C(c2c(CC)ocn2)=O)CC(NC(c2cccc(CC)c2C)=O)CC1(CC)CC C(COCCO)(CC(=O)NC(C)CCCO)NS(CC)(=O)=O.C(=O)C(C)(C)C c1(OCC)nc(C)ccc1C.C(Cc1cccs1)(CC=C)NC(=O)NC1CC1OCC CC(C)CC(C)C(C(=O)NC(C)C)N1CCCCC1CN1CCOCC1 CCC(C(=O)NCCOCCOCCNC(=O)C(C)C1CCCO1)C(C)O c1(C(N2CC3C(CNC(C4C(C(N)=O)C4)=O)(C3)C2)=O)cc2nccn2c(O)n1 c1(OC)ccc(C(=O)NC(C2CCCC2)CNC(=O)CNC(=O)NC)cc1 Cc1nncn1NC(=O)CC(C(C)(C)C)NC(c1nnc(S)n1C)=O CC1CN(C(c2nccs2)=O)CCC1NC(=O)C(F)=C1CCC1 c1(C(C2CC(F)C2)NC2CN(C(=O)OC(C)(C)C)C2)ncccn1 C#CC1(O)CCCN(C(=O)C(CNC(=O)CSC(F)(F)F)C(C)C)C1 c1(C(=O)NC2CCN(C(c3c(CC)non3)=O)C2)cc(F)cc2c1CCC2 Cc1ccc(F)c(S(=O)(=O)N2CCc3ccccc3C2)c1.N1(CC)C2CCC1COC2 CC1CCc2nc(C(N3CCC4(C3)CN(C(C3CCC(F)(F)C3)=O)C4)=O)cn2C1 c1(C(=O)NCCN(C(=O)C=Cc2cnn(C)c2)C(C)C)nc(=N)cc[nH]1 Cc1c(-c2cn(CCCC(=O)NCCc3ccco3)nn2)cccc1F CC(C(=O)NCC1CN(C(C2(F)CC3(CCC3)C2)=O)CCCO1)S(N)(=O)=O N1(c2cc(NCCc3ccc(C(F)(F)F)cc3)ncn2)CC2CCCC2C1 C1(CNC(c2cccc(C)c2)=O)CC(C)(C)CCC1NC(c1nc(C)c(C)s1)=O CC1(C)C(NC(c2cc(CN(C)C)on2)=O)CCN1C(c1csc2nnsc12)=O c1(C(=O)NC(C)CNC(C2(F)C3CCCC23)=O)ccc(Cl)c2ccccc12 S(=O)(=O)(c1ccc(O)c(-c2nn[nH]n2)c1)N1C(C)CC(O)C1 N1(C(C(CC=C)NC(=O)CCc2cnc(C)o2)=O)CCN(C)C(C)C1 CC(C)CCC(=O)NCC(C)(O)CNC(=O)CCOC1CCCC1 c1(C(=O)NCCC(C)NC(C)=O)cn(CCN2CCSCC2)nn1 c1(C(=O)NCC(n2cc(C3CC3C)nn2)C)ccc(C(=O)O)cn1 C(=O)(C1SCCc2ccccc21)NC(C)(C)CCNC(C1CC2(CC2)CO1)=O N1(C(CC(C)(C)O)=O)CC(NCc2c(O)cccc2O)CC(F)C1 Cc1sc(N)c(C(N2CC(NC(=O)C(F)CC3CCC3)C3(CC3)C2)=O)c1C C1(C(N(CCN(C(C(CC)(C)O)=O)C)C)=O)Cc2ccc(F)cc2O1 c1(NC(c2n(CCCC)nnn2)C2(N(C)C)CCCC2)cc(OC)cc(OC)c1 C1(CNC(c2cc(C)oc2C)=O)CC(C)CN(C(C2CCCCCN2C)=O)C1 c1(OC(C(=O)NCCN(C(C(F)=CCC)=O)CC)C)ccc(F)cc1 n1(CC)ncc(C(=O)NC2CCCCC2CNC(C2(c3ccsc3)CC2)=O)c1C C12(COC)CC(CNC(c3ccc(F)c(F)c3)=O)(CN1C(C1CCC(=O)N1)=O)C2 n1(CC(N2CC(C(C(=O)NC(C3CCC3)C3CCC3)OC)C2)=O)cnnc1O Cc1cc(O)ccc1-c1cn(C2CN(C3CCC(=O)N3C)C2)nn1 c1(C(=O)NCC(C2CCCN2c2ncnc(=N)[nH]2)(C)C)cc2n(n1)CC(F)C2 c1(C(N2CCCC(C(=O)NC3C(C)(C)CCC3)C2)=O)cnc2ccnn2c1 CCC(CC)CC(=O)N1CCCC1C1CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 N1(C(C(C2CCC2)OCC)=O)CC(CNC(c2cn(C)cc2C)=O)OC(C)(C)C1 C=C1COc2c(C(N3CCC(C)(CNC(c4cc(O)nn4C)=O)C3)=O)cnn2C1 C1(NC(C2(COC)CC(=C)C2)=O)CC(C(=O)NCCc2cc(C)no2)=CC1O Cc1ncccc1-c1ccc(CN=C(NC(C)C2CC2)NC2CC2C)cc1 c1(C(N(C(CNC(C(CC=C)(C)C)=O)C)C)=O)cnc(O)n(C)c1=O c1(N(C)Cc2n(C(C)C)cnn2)nc2ccccc2nc1N1CC2CC1C2 CCCCCCC(C)C(=O)N(CCC(N1CCC2C(C(N)=O)C2C1)=O)C(C)C Cc1cnc(CC(=O)NCC2CC23CCC3)o1.c12nocc1NC2=O Cc1ncnc(C)c1C(=O)N(C)CC1CCN(C(C2CCS(=O)(=O)N2)=O)C1 C1(NC(c2ccc(CCC)[nH]2)=O)CN(CC(O)CC(F)(F)F)CC(C)(C)C1 c1(OC)ccc(CNC(=O)C(=O)Nc2ccc(C(C)(C)C)cc2)cc1C(C)C C(=O)(CCCCCS(N)(=O)=O)N1CCN(C(c2[nH]n(C)c(=O)n2)=O)C(CO)C1 Cc1ccc(C=CC(N2CCCCC2CCCNC(=O)C(C)(O)C2CC2)=O)cn1 CC(C)(C)C(CO)C(=O)NCC1(C(N2CCC3(CCC3)CC2)=O)CCC1 C(=O)(CCCC(=O)N1CCCCC1C1CCCN(C(C2(C(C)=O)CC2)=O)C1)NC N1(C(C2(NC(C(C=C)C)=O)CCOCC2)=O)CC(C)C(O)C(C)C1 c1(CNC2CCC(C(=O)Nc3c(OC)nc(C)cc3)C2)c(F)ccc2occc12 c1(C(=O)NC(C(C)NC(c2cn(CCCF)nn2)=O)C)cnccc1Cl C1(N(c2nc(C)cc(C)n2)C(C(C)NC(CC)=O)=O)CCNCCC1C c1(C(=O)NCC(CNC(c2c(CC)c[nH]c2)=O)OC)cc2c(C(C)C)nn(C)c2s1 c1(OC)ccc(CCC(N2CC3(CCN3C(c3ccc(O)cn3)=O)C2)=O)cc1C C(=O)(CC(CC)CC)N(C1CCN(C(COCC(=C)C)=O)CC1)CCOC C1(C(=O)NC2CC(NC(C(CN(C)C)N(C)C)=O)C2)COC2(CCC2)C1 CC(C)C(F)(F)CC(=O)NCCOCCCN(C)C(c1csnn1)=O c1(C(N2CCC(C(C)(C)NC(C(CC)O)=O)C2)=O)csc2cccnc12 O=C(C(F)(F)C(F)(F)F)NC1CC(Nc2cc(CC3CC3)ncn2)C12CCC2 C1(C(N(C(CNC(C2CC(O)(C(F)(F)F)C2)=O)C2CC2)C)=O)CCC2(CCC2)C1 c1(C(N2CC(C)C(NC(=O)CN3CC(=O)NC3=O)C2)=O)cc([N+](=O)[O-])cnc1N C1(C(=O)NC2CC(C#C)C2)CSCCN1C(C1CC(C2CC2)C1)=O Cc1cc(O)c(C(=O)NCC2CCCN(C(=O)COc3ncccn3)CC2)nn1 c1(OC)cnc(F)c(C(=O)N(CC(C)(C)NC(=O)Cc2cnccc2C)C)c1 c1(C(=O)NC2CC(NC(C3CC4(C3)CC4(F)F)=O)C2)ccc2c(c1)CCCC2 Cc1ccc(C(=O)NCC2CCCCC2NC(=O)C2=CCSC2)cc1N C(=O)(C#CC1(C(F)(F)F)CC1)NC(C)CCCCNC(=O)C=Cc1ccn(C)c1 CC(CN=c1[nH]c(N2CCC(CF)C2)nc2c1CSC2)c1cccc(Cl)c1 C1(CNC(=O)NC2(C)C(C)(C)C2)(CSC)CC(F)(F)C1.[SH](C)(=O)=O c1(C(C)NC(N2CCCCC2Cn2ccnn2)=O)cccc(Cl)c1Cl N1(C(c2n(OC)cnc2C)=O)CC2(CC(C(=O)Nc3cc(C)cnc3O)CO2)C1 CC1CC(C(N)=O)CN(C(=O)CCCc2cc(F)ccc2F)C1 c1(CC)ccccc1C(=O)NCC(=O)NC(C(=O)N(CCOC)C)C1CC1 Cc1cc(C(=O)NCC(C)(O)CNC(C2COCCO2)=O)c(N)c(Cl)c1 c1(OC)ccc(NC(=O)C(C(C)(C)C)N2C(=O)CCC2=O)c2ncccc12 CCCCCC(O)CC(=O)N1CCCN(C(=O)COc2cccnc2O)CC1C FC(F)C(CN=c1[nH]c2c(c(=NC3CCN(C4CC4)CC3)[nH]1)CCCCCC2)NCBr Oc1cc(C(F)(F)F)ccc1CN1CCSC2CCCC12 c1(CC)ccc(-c2nc(C(F)CF)n(-c3ccc(-c4ccccc4)cc3)n2)cc1 C1(N(C)C)(C(=O)NCCC2(CNC(C3OC4CCC3C4)=O)CC2)CCCSC1 Cc1cc(C(N)=O)cc(C(=O)NC2CCOCC2NC(=O)CC2CCOC2=O)c1 CCCC(CCNC(=O)C#CCNC(C1CC1CC(C)(C)C)=O)C1CC1 C1(OC)CC(CNC(=O)CCOc2cccnc2)N(C(=O)C=C2CCC(C)C2)C1 N1(C(C2(CCCC)CC2)=O)CCOCC(CNC(C23CCC(CC)(C2)OC3)=O)C1 C1(F)(CNC(Cc2nn(C)c(Cl)c2)=O)CCCN(C(=O)C2=CCCCCC2)CC1 Cc1ccc(C(=O)CCC(N2CCC(NC(=O)CC3CCOC3)CC2)=O)cc1 C(CC(C(=O)Nc1ccc(C2CC2)nc1)NC(=O)COCC(F)F)=CC C=CC1OCCC1C(=O)NC(C1CCN(CC(C)CC)CC1)C c1(-n2c(C(=O)NCC3C(NC(=O)COC4CCOC4)C3)cnn2)ccccc1Cl C1(NC(c2ocnc2C2CC2)=O)CCCCN(C(c2cc(F)cc(F)c2)=O)C1 c1(C(N(C)CC2CCN(C(=O)OC(C)(C)C)C2)=O)ccccc1S(=O)(=O)C(F)F c1(C(=O)NC2CCCC(NC(Cc3cc(C)no3)=O)C2)cc2sc(Cl)cc2s1 C1(NC(c2cc(Br)co2)=O)CN(C(C2(CF)COC2)=O)CC1CO C1(NC(c2ccc(OCCC)cc2)=O)CC(NC(=O)C(F)C2CCC2)C12CCC2 C(=O)(C(C)C(O)CC(C)C)NCC1(F)CN(C(c2ccc(C)nc2)=O)C1 CCCCCC(CC)C(=O)NC1CN(C(c2ccnn2CC)=O)CC2CC12 c1(C(N2C(CNC(C(CC(C)C)C)=O)CC3(CC3)C2)=O)cc(Cl)cc(Cl)c1N C1(C(N2CC(C(C)NC(CC(=O)NCC)=O)OCC2)=O)(CF)CC2(CCC2)C1 C1(NC(=O)CC2COCCO2)CN(C(C2(n3cncn3)CC2)=O)CCC12CCC2 C1(C(C)C)CN(C(=O)Cc2ccc(C#N)nc2)CCCN1C(=O)CC1CCOC1 C1(N)CN(C(C2CC23CCCC3)=O)CC12CC2.Cc1nc(CC=O)sc1C Cc1ccc(C)c(OCC(C)NC(=O)C(=O)N(C)Cc2nccn2C(C)(C)C)c1 N1(C(c2c(COC)cco2)=O)CC2CC2C1C(=O)N(C)CC1CCCCO1 c1(NCC2CC2)ccc2c(c1)OCCN2C(N(CCC(C)OC)C)=O.C(C)(C)(C)NC=O c1(C(=O)NCC(C(=O)NC(C(C)C)c2nc[nH]n2)OC)c(C)n[nH]c1C C1(CC(=O)NCC2N(C(c3cc(C)no3)=O)CC2)CC2(CCC2)C1 c1(OC)ccnc(C(N2CCC(C)(c3cn(CCCCF)nn3)C2)=O)c1 c1(NC(C2CCCN(Cc3csc(NC(=O)OC)n3)C2)=O)cc(F)c(F)c(F)c1 N(C(=NCCCF)NCC1(C)C=CCCC1)C1CCC(SC)C1 C(=O)(CC(C(F)(F)F)n1cccn1)NCC1(CNC(c2c(C)cccn2)=O)CC1 N1(CC)N=C(C(=O)N2CCN(C(=O)CC(C)P(C)(C)=O)CC2CCO)CCC1=O c1(C(N2CC(CCNC(C(COC)(C)C)=O)OCC2)=O)ccc2cnnn2c1 c1(CC(=O)NCC2N(C(CCC(=C)C)=O)C3C(C2)C3)ccc(C)c(C)c1 C(C(C)(C(=O)NCCCCC1CC1)NC(=O)C(F)CC1CCOC1)SC N1(C(COCCC)=O)CCC2(CCOCC2)C(NC(c2ccn(C(F)F)n2)=O)C1 C1(C(N2CCCC(C)(CNC(CSCCN(C)C)=O)C2)=O)CCC2(CCC2)CC1 c1(N(CCCCN(C(=O)CC2(C)CC2)C)C)c(C#N)cnc2ccccc12 n1(CCC)cccc1C(N1CCCC1CCCNC(=O)CCc1cccnc1)=O N1(CC)CCCCC1C(=O)NCc1ncccc1C(=O)NC1CCSC(C)C1 N1(C(c2c(C)cn(C)c2)=O)CC2CN(C(=O)CCC(N)=O)CC12 c1(OC)csc(C(=O)N(C(C)CNC(=O)C(C)(C)c2cc[nH]n2)C)c1OC C1(CCOC(C)(C)C)CCCN1C(C1CC1F)=O.C1CC(=O)N1 N1(C(C(CC)=CC)=O)CCN(C(=O)CC2CC(=O)NC(=O)C2)CC1CC C=C(C)CCCC(=O)N1CCCC(CCC)(NC(c2cncc(OC)c2)=O)C1 CCC(CC)C(=O)N1CC2CC2(NC(c2cnn(CC3CCCO3)c2)=O)C1 CCN=C(NCCCc1snnc1C)NCc1cnnn1-c1ccccc1 CC1CN(C(C2(Oc3ccccc3)CC2)=O)CC1NC(C1CC12CCCC2)=O C1(NC(c2ccc(C)nc2N)=O)CC2(CCC(NC(C3(C)C=CCC3)=O)CC2)C1 CC(CCCCNC(C1CC1C#N)=O)NC(=O)CC1(C)CC(F)(F)C1 c1(OCC(=O)NCC(CCNC(C=C2CCN(C)C2)=O)O)c(F)cccc1F c1(OCC)ccc(F)cc1C(N1CCN(C(=O)C=Cc2ncc[nH]2)C(CF)C1)=O CSC=CC(=O)NCC1(NC(c2scnc2C2CC2)=O)CC1 c1(OC)cnc(Cl)c(C(=O)NCCN(C(=O)C(C)n2cccc2)C2CC2)c1 c1(C(=O)NC(CNC(C(F)=CCC)=O)Cc2ccccc2)nn(C)cc1N C(=O)(CCN(OC)C(=O)c1nc(Cl)oc1C)N1C(CCOC)CCCC1 C1(C)(c2nc(CC)[nH]n2)CCN(C(c2cnn(C)c2)C(=O)NCCCC2CC2)C1 c1(C(N(CCC(=O)NC(CCC)C2CCCC2)CCCO)=O)cccc(Cl)c1 c1(CCNC(C(C2CCN(C(C3CS(=O)(=O)C3)=O)C2)C)=O)cnn(C)c1 C1(NC(C2CC2(F)Cl)=O)CN(C(c2ccc3c(c2)CCO3)=O)C2(CCC2)C1 C=C(C)CC(=O)NC1CC1CNC(c1csc(COCC)n1)=O C1(NC(Cc2nc(C)sc2)=O)CC2CC(C1)N(C(c1cnn(C(C)C)c1C)=O)C2 N1(C(CCN(C)C)=O)CCC(c2cnn(C)c2)CC1.c12cn(C)nc1CNC2=O N1(C(=O)CSCC2CCCCO2)CCC2(CC1)CCN(C(C1CC(F)C1)=O)CC2 C1(NC(c2c(OC)coc2)=O)CC(O)CN(C(=O)CC23CC(C2)C3)C1 c1(OC)ccnc(O)c1C(=O)NCC1(NC(C2CCNC2=O)=O)CCOC1 c1(C(N2CC(C(C)NC(C3C=CCS3)=O)C2)=O)ccc(F)c(Cl)c1F c1(N2CCC(C(C)C)CC2)nc(=NCCN(C)S(=O)(=O)N(C)C)[nH]c2ccsc12 N#CC1CCN(C(c2nc(Br)ccc2Cl)=O)C(c2ccccc2)C1 C12(NC(C(C)N3CCCC3)=O)CCCC(NC(=O)CSS(C)(=O)=O)(C1)C2 c1(OC)cc(S(=O)(=O)N2CCCC(CNS(=O)(=O)c3ccncc3)C2)ccc1Br C(C)(C)(CC(F)C(=O)N(C)CC1(C)CC1)NC(C(N1CC(C)C1)C)=O n1(CC=C)cccc1C(=O)NCCCN(C(=O)C(C)CC1CC1)C CN1CC=C(CC(=O)N2CCC(F)CC2C(=O)NCCCSC(F)F)CC1 c1(COC)c(C)nn2ccc(C(=O)N(C3CCCSC3)CCO)nc12 c1(CN2CCN(C(c3ccc(C)c(Cl)c3)=O)C(C#N)C2)c(F)ccc2[nH]ccc12 C1(c2ncc(C(=O)OC)c(=O)[nH]2)CCCN(N2CCC3C(CCC3CO)C2)C1 N1(C(c2c(COC)cc[nH]2)=O)CCOC(CCCNC(C2CCC(F)(F)C2)=O)C1 c1(-c2nc(CN3CCC(C(=O)O)(CC)CC3)on2)cccc(S(C)(=O)=O)c1 c1(CC(=O)NCC2N(C(CC3(NC(C)=O)CC3)=O)CCSC2)cccc(O)c1F C1(NC(C(CCSC)O)=O)CC2CN(C(c3ccn(CC(C)C)n3)=O)CC2C1 N(S(=O)(=O)N1CCC(OC(F)F)CC1)(c1cccc2ccccc12)CC N1(C(C2(F)CCN(Cc3cc(F)cc(Cl)c3)C2)=O)CCc2cccc(Cl)c2C1 C1(CC)C(NC(=O)CN(C)C(N)=O)CCN1C(c1ccc(NC(C)=O)cn1)=O N1(C(C=C(C)C)=O)CC2CCN(C(c3ccc(C)c(CO)c3)=O)C2C1C C1(NC(CC(C(=O)OC)C)=O)CCC2(CC1)CC(NC(=O)Cc1csc(C)n1)C2 c1(C(N2CCCC2c2ccc(C)s2)C(=O)NC(C(=O)OC)C)coc(C)n1 C1(C(=O)O)CCC(c2ccc(C(N3CC4CC4C3)=O)cc2)CC1 C(=O)(C(C)(C)CCC#N)N1CC2(CC(NC(C(C)NS(CCCC)(=O)=O)=O)C2)C1 N1(C(CCSC)=O)CCC(CNC(c2oc(-c3cnn(C)c3)nc2C)=O)CC1C N1(C(CCc2ccc(=N)[nH]c2)=O)CCC2(CC1)CC(NC(c1coc(Cl)n1)=O)C2 N1(C(=O)CC(F)(F)Cl)CCN(C(C2CCCCC2F)=O)CC12CC2 C1(C(=O)NC(C2CCN(C(c3c(CC)csc3)=O)C2)(C)C)CC(C)(C)CCO1 CN1N=CC(CC(=O)N(CC(=O)NCC2CCC3(CC3)C2)CC2CC2)C1=O c1(SCC)nccn1C(C)CC(=O)NCCCCCN(C(=O)C(CC)N(C)C)C C(CC(C)(C)C(=O)N1CCOCC(NC(C2CC2C(F)(F)F)=O)C1)SC c1(OC)cc(C(N2C(CNC(=O)COCCF)CC3CC23)=O)cc2c1OC(C)C2 Cc1cscc1C(=O)NC1CCC(NC(C2CC(CC3CC3)C2)=O)C1 N1(C(c2ccc(C(C)C)s2)=O)CCC(N(C)C(c2coc(CO)n2)=O)C(C)C1 O(C=C(C#N)C(=O)N1CC(CNC(=O)C(c2ccc(Cl)c(F)c2)O)C1)CC N1(C(CCC(=O)NC)=O)CCC2(CCC2NC(c2cn3cc(C)sc3n2)=O)CC1 C(=O)(C(C)(CO)NC(=O)Cc1cccs1)N(C)Cc1nc(C)[nH]n1 C(=O)(C(C)(C)CC(C)(C)C)NC(CCNC(CCC(=O)NC)=O)(C)C C(=O)(C1=CCCSC1)NCCN(CC(C)O)C(c1n(CC#C)ccc1)=O CC(C)S(=O)(=O)C(C)C(=O)N(C1C2CN(C(=O)C=C3CCSCC3)CC12)C CC1CCN(C(=O)CCc2ccc(F)nc2)CCN1C(C1CC1C1CCCO1)=O C(=O)(CCC(=O)NC(C)(C)CC=CC(=O)NC1(CC)CCOC1)NCCC CCCCC(F)C(=O)N1CCCC1C(=O)NCc1ccoc1C N1(C(C2CC(C(C)C)OCC2)=O)CC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 N1(C(C2C(CNC(c3cc(C)c(C)o3)=O)OCC2)=O)CC=C(C(C)(C)C)CC1 C12CCC(CC1)CNC(=O)CN2C.C1(CC(=O)C2CCC2)CC2CCC1O2 C1(F)(CNC(c2ccc(Cl)cc2C(F)F)=O)CCCN(C(C2CCCC2)=O)C1.SCC c1(OC)cccc(=Nc2cccc(C(N3CC4(C)CC3CCO4)=O)c2)[nH]1 N1(C(c2c(C)noc2)C(=O)Nc2ccc(F)cc2)CCC2(CC1)CC(C1CC1)=NO2 N1(C(CCC2C(C)=NNC2=O)=O)CC2CC1CN2C(c1cnncc1C)=O N1(C(C2COCC(C)O2)=O)CCC(C(=O)NCCc2cc(O)no2)C(C)(C)C1 C(=O)(C(C)C(C)NC(=O)CC1CC(=O)C1)NC1(c2nc(C)on2)CC1 c1(C(=O)NC2C3(CN(C(c4cccc(N)c4O)=O)C3)CC2)cc2ccccc2s1 c1(C(=O)NCC2C(NC(c3cc(CC)nn3C)=O)CC2)cc2cc(F)ccc2o1 N(C1CCOc2cc(F)ccc21)NC(C1CC1C1CC1)=O.C123CC(C1)(C2)C(=O)N3 c1(CNC(CN(C(=O)CSCCC#N)CCC)=O)cn(C)cn1 c1(CCNC(=O)NC2CC(C)OCC2)cc2ccccc2o1 C(CCC(C)C(=O)NCC=C1CCN(C(c2cc(O)cc(Cl)c2)=O)CC1)OC C1(C(N(CC(CN(C(CCC=C=C)=O)C)O)C)=O)COCCC1(F)F Cc1cc(O)nc(C)c1C(N1CCCCC(NC(=O)CSCC(F)F)C1)=O c1(C(=O)NCCC2CCN(C(C(CC)NC(C)=O)=O)C2)ncnc2c1OCCO2 n1(CC)cc(Cl)c(C(=O)NCCCCC(C)NC(=O)CC(C)c2cnn(C)c2)n1 C1(CNC(C2(C#C)CCC2)=O)CCC2(CN(C(c3cc(C)c(Cl)c(N)c3)=O)C2)O1 CC(CC1CCCC1)C(=O)NCC1(CNC(C2CCC(CO)O2)=O)CC1 c1(OC)ccc(CO)cc1C(=O)NC1COCC1C(=O)NC1CCC(O)C1 C12(NC(CCC)=O)CCC(CC1)N(C(=O)C(C)(C)n1ccc(C)n1)C2 CCC(C)C(C)C(=O)NCCCN(C(=O)CCSC)C(C)C c1(N2CC(C(=O)NCc3cocn3)C(O)CC2)ncnc2sccc12 C1(c2c(C(N3CC(OCC)C3)=O)c[nH]n2)CCCCN1C(=O)CC(C)C1CC1 N1(C(c2ncoc2-c2cccc(F)c2)=O)CCC2(CC2COBr)C1 C1(C(C)C)CCC(C(=O)NCCCCNC(c2cc(C(F)(F)F)nn2C)=O)CC1 N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCC(C1)N(C(c1ccc(F)c(CO)c1)=O)C2 c1(NCC(C)N(CCCc2cn(CCOC(C)=O)nn2)C)ccc(F)cc1Cl N1(C(c2cnn(C)c2N)=O)C(C(=O)NCc2nc(CO)n[nH]2)CC2CCCC12 N1(C(C(C(CC)O)(F)F)=O)CCCC(N=c2nc(C(=O)C(C)(C)C)[nH]s2)C1 CC(C)CCC(O)C(=O)NC(CC(=O)NC(C)C(C)(C)C)C(F)F c1(OC)ncc(C(N2CCC(CCO)C2)=O)cn1.C(=O)(COCC(=O)NCC(C)C)OC C1(C(N)=O)(NC(c2scc(C(C)N(CC(F)(F)F)CC3CC3)n2)C)CCNCC1 Cc1nc(C(F)(F)F)ccc1C(=O)NC1(CNC(=O)C(F)(F)F)CC1(C)C N1(C(C(CN(C)C)c2ccccc2)=O)CCCC(N(C(=O)C=CC2CC2)CCO)C1 C1(NC(c2ccn(C)c2)=O)C2CC(NC(=O)CC3COCC3(C)C)CC12 N1(C(C2(C(=O)N(CCC(F)(F)F)CCO)CC2)=O)CCCC(c2ccccc2)CC1 CC1CCN(C(=O)CC2COC(=O)C2)CC1NC(C1CCC(C)CC1)=O CC(CCCCCO)NC(C1CC2CCC1N2C(c1cc(=N)[nH][nH]1)=O)=O CC(O)C(C)C(=O)N1CCN(C(C)CNC(=O)CSc2cn[nH]c2)CC1 c1(CCNC(=O)NC(c2ccc(F)c(F)c2)CC(=O)NC)c(C)cc(C)cc1C N1(C(C(C)N(C(c2cn(CC)nc2)=O)C)=O)CCC2(CCOC2)C1 N1(C(C(C)NC(=O)OC)=O)CCC(C(C)C(=O)N(c2cn[nH]c2)CCO)C1 c1(C(N2CC(C)(NC(CSCCC(C)C)=O)C2)=O)coc(S(N)(=O)=O)c1 c1(NCc2c(C)nc(C)[nH]2)cnn2c1OCC(C(=O)O)C2 c1(SC(C)C)ncccc1C(=O)NC(C)C(CO)NC(c1cn(C)c(O)n1)=O c1(C(=O)NCC2(CO)CCN(C(CC3CC(C)C3)=O)C2)ccc2c(c1)OCC2 N1(C(COCCOC)=O)CC(NC(c2ccc(F)c(CO)c2)=O)CC12CCOC2 C12CCN(CC1)C2=O.C(=O)(CCCN1CCOC1=O)NC(CC)(C)C C1(=CC(N2C(C)CC(NC(c3n(CCC)nc(C)c3)=O)C2)=O)CCC(C)(C)CC1 C(=O)(CCCCCOCC)NCC(C1CC1)NC(c1c(CC)nc[nH]1)=O O=C(C1=CC2CC=CCC12)NCCNC(c1cnc2sccn12)=O c1(C(=O)NC(CNC(c2c(C)coc2C)=O)(C)C2CCC2)ccc(S(C)=O)cc1 C(=O)(C1=NOCC1)N1CCC(CCNC(C(C)c2ccon2)=O)C1 c1(CC(=O)NC(C2CN(C(c3cnc(COC)s3)=O)C2)C)ccc(F)c(F)c1 C1(C(=O)Nc2c(CC)csc2)(CC)CCCN(C(=O)C(F)(F)C(F)F)C1 N1(C(C=C(CCC)C)=O)CCCCCC1CNC(c1cc(OC)ccc1C)=O C1(NC(Cc2ccc(C)s2)=O)CC(C(=O)N2CCCC2C2(N(C)C)CC2)=CC1O CC1CN(C(C2CC(F)(CO)C2)=O)CCN1C(c1ccc(F)c(Cl)c1)=O c1(C(N2CCC(CCNC(C(C)C(F)F)=O)C2)=O)cc(C(N)=O)ccc1F C1(COC)(NC(C2CC2(Cl)Cl)=O)CCCN(C(c2ccc(NC3CC3)cc2)=O)C1 c1(C(=O)NCC2CCN(C(C(CC)(F)F)=O)CC2)cc2ccccn2n1 N1(C(c2ncc(NC)nc2)=O)CCC2CN(C(c3cncc(C)c3)=O)CC2C1 c1(SCC(=O)NCC(C2CC2)NC(C(c2cccnc2)OC)=O)ccoc1C c1(C(N2CC3C(CNC(CC=CCC)=O)(C3)C2)=O)ccc2c(c1)CCC2(C)C N1(C(C(C(C)C)CO)=O)CC2CC(NC(C3CC3(c3ccccc3)C)=O)CC1C2 C(C(=O)NC1CC(CO)C1)(C1=CCC2CC2C1)NC(=O)OC(C)(C)C Cc1ccc(Cn2nc(-c3cccc(C)c3)nc2CCc2ccc(F)cc2)cc1 c1(C(F)F)cccc(OC)c1.n1(CC)nnnc1CNC(c1cn(C)nn1)CC C(N=c1[nH]c(=NCCCOCCO)[nH]c2ccccc12)c1c(OC)ccnc1O C1(F)(C(N2C(C(=O)OC)CC2)=O)CCN(C(=O)C=CCO)CC1 Cc1c(C(N2CCCC2C(C)(C)NC(=O)C2=C(Cl)CC2)=O)n[nH]c1C1CC1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CSc2ccc(Cl)nc2)C(C2CCC2)C1 Cc1nc(CCC(N2CCCC(CNC(C3CC(F)(CO)C3)=O)C2)=O)cc(O)n1 c1(C(=O)NC2C(CNC(C3(C)C=CCCC3)=O)COC2)cc(O)cc(=O)o1 CCC(CC(=O)N1CC(CC(=O)N(CC(C)O)CCO)C(C)C1)SC C#CCCC(O)C(=O)NCc1ccccc1CNC(c1ccccc1F)=O N1(C(CSC(C)C)=O)CC(CNC(=O)CCCNC(=O)C(C)(C)C)CCC1C C1(C(=O)NC(CCN(C(C(C(CC)O)C)=O)C)C(C)C)CCc2nncn2C1 c1(CCC(=O)OCc2ccc(C3CC3Cl)o2)cccc(Br)c1 N1(C(C(C)C#N)=O)CC(CNC(C2(c3ccc(Cl)nc3)CCC2)=O)C2(CC2)C1 c1(OC)ccc(NNC(=O)CSC)cc1-c1scc2c1CCC2 C1(C(N(CCOCC)CC)=O)CCC(CNC(=O)CC(C)n2ccnc2)CC1.C1CC1 n1(CC(=O)NCCNC(C=C(CCC)C)=O)ncc2ccc(Br)cc2c1=O N1(C(C(F)=C(C)C)=O)CCc2sccc2C1CNC(=O)CCOC1CCCC1 c1(C(N2CCC(N(C(=O)CCc3ccncn3)C)C2)=O)cc(N)ccn1 C(=O)(CC1=CCOCC1)N1C2CC(C(=O)NCC(CCCCC)O)(OC2)C1 N1(C(C(C2CCCN(C(Cc3c(C)cccc3)=O)C2)(C)C)=O)CC2CCOC2C1 C(=O)(CN=c1cc[nH]cc1)N1CCC(OCCNC(c2n[nH]c(C)c2Cl)=O)C1 C1CCCCC(=O)N1CC.C1(CC)CC1C(=O)NCCOC.C(=O)(COCCO)N c1(CC(=O)NCC2C(NC(c3nc(OCC)oc3)=O)COC2)cc(F)ccc1F c1(OC)ccc2nc(C)nc(N3CCCC3C(=O)NCCC3CCCO3)c2c1 CN1CCCC(CC(N2CCC(C(=O)N(C)CCF)(N(C)C)C2)=O)C1 C1(COC)(NC(C2CN3CCC2C3)=O)CCN(C(c2ccncc2F)=O)C1 CC1CN(C)CCC1NC(C1CNC(=O)CN1C(c1ccc(CC#N)cc1)=O)=O c1(C(=O)NCC2(O)CC(CNC(C3(C)CCOC3)=O)C2)cc2ccc(Cl)cc2[nH]1 CN1CCC(C(=O)NCC(C)(CO)NC(c2cnc(Cl)s2)=O)c2ccccc21 C1(C#N)(C(=O)NCC(N2CCN(C(C(CC#C)(C)C)=O)CC2)=O)CCN(C)CC1 C(=O)(C(F)C(C)CC(C)(C)C)NC(CCOC)CNC(=O)CN1CC(C)(OC)C1 N(C(=NCC(=C)C)N1CCC(c2ccccc2F)C1)CCOCCC#C c1(C(=O)OC)[nH][nH]c(=NC(=O)N2CCN(CCO)C(=O)C2)c1C1CC1 C=CCCC(=O)NCC(O)C(=O)NC(COC1CC1)CO N1(C(C2N(C(COC)=O)CCCC2)=O)CCN(C(C2CC(=O)N2)=O)CC1CO c1(OC)cc(CNC(C2CC(C)N2C(C2(CO)CC2)=O)=O)ccn1 c1(C(N2CC(N(C(c3c(C)ccnc3)=O)C)C3(C2)CC3)=O)cc(O)cc(N)c1Cl c1(C(N2CCCC(C)(CNC(CC3CC(OC)C3)=O)C2)=O)ccc(S(C)(=O)=O)[nH]1 C1(NC(c2c(C)[nH]cc2)=O)CN(C(c2oncc2C)=O)CC1C1CC1 N1(C(C2CN(Cc3ccc(C)s3)CC(F)C2)=O)CCc2nc[nH]c2C1 c1(C(=O)NC2C(C(=O)Nc3c(C)ncc(C)n3)CCC2)cc([N+](=O)[O-])ccc1C c1(C(N2CC(NC(=O)C(F)=CCCF)CC(C)(C)C2)=O)ccc([N+](=O)[O-])c(N)n1 c1(C(N2CCN(C(C3CCC(C)N3C)=O)CC2CO)=O)cnc2[nH]ccnc1-2 c1(C(N2CC(c3cn(CC(F)(F)CO)nn3)C(O)C2)=O)cc(F)ccc1F C1(NC(CCC2CC(OC)C2)=O)CC2CCC1(NC(=O)Cc1nc(C)sc1C)C2 OC1COCCC1C1CCC1.c12cccc(c1)-n1cc-2nn1 CN1C2CCC1CC(CC(=O)NC1(CF)CCN(C(C34CCC(CC3)C4)=O)C1)C2 C(=O)(C(CC(F)F)N(C)C)N(CCNC(C(CC)OC)=O)CC1(COC)CC1 C1(C(=O)NC(Cn2ncc(C)c2)C)(CNC(=O)CSCC(F)F)CC12CCC2 C(=O)(N=c1nc2ccc(Cl)cn2[nH]1)c1c(CC(C)(C)C)c(F)ccc1 c1(C(N2CC(CNC(c3ccncc3I)=O)OCC2)=O)cc(Br)ccc1Br c1(NCC)cc(NCCNC(c2cccs2)=O)nc(C(F)(F)F)n1 c1(NC(c2nc(NC(c3scc(C)n3)=O)sc2)=O)cnc(C)c(F)c1 CC1(C)CC(C)N(CC(C(=O)C(C2CC2)C2CC2)=O)C1.c1(CN)ccccn1 c1(CC)cccc(OCC(=O)NCCCC2CN(C(c3cccs3)=O)CCO2)c1 C1(NC(NCC(CCCC)CC)=NCC)CCSC2(CCC2)C1 C(CCCCCNC(=O)Cn1cc(Br)cn1)N(C)C(c1ncn(C)n1)=O CCC(C)C(C)(O)CNC(C1(CNC(c2nocc2Cl)=O)CC(C)(C)C1)=O c1(OC(C(N2CCCC(NC(c3c(OC)ccs3)=O)C2)=O)C)cccc(Cl)c1Cl N1(C(c2cnc(C(C)(C)C)[nH]2)=O)CCC(C)(CCNC(C2CNC(=O)N2)=O)C1 Cc1ccc(C)c(OCCC(N2CCC(C)(NC(C3CCOC(C)C3)=O)C2)=O)c1 c1(C(N2CC(C(C)NC(=O)CC3CCOC3)OCC2)=O)cc(C#N)ccc1N C1(COC)CC(CNC(C2CCCN(C)C2)=O)N(C(c2sc(C)cc2C)=O)C1 N1(C(=O)Nc2c(CC)ccc(CC)c2)Cc2[nH]nc(-c3ccc(OC)cc3)c2C1 N1(C(C2(C)CCC2)=O)CCC(CO)(CNC(=O)CCCc2ccncc2)CC1 C(=O)(C(C(C)NC(=O)CCc1cccnc1)C(C)C)NCC1(OC)CC1 N1(S(CC=C)(=O)=O)CCN(CC)CC1.C(CCCCCC)OCCN1CCCC1 C(=O)(C(F)CC(C)(C)NC(=O)CCC1CCOC1)NC(C(C)C)C1CCC1 CCC(C)C(C(=O)N(C)OCC(F)(F)F)NC(=O)CN(C)C.C(C(=O)OC)S CC(C)C(C#N)C(=O)N1CCCC(F)(C(=O)NC2CC(C3CCC3)C2)C1 C1(NC(COCC(C)C)=O)CC2CCCC(C1)N2C(=O)Cc1csnn1 CCCC(C(O)C(=O)N(C1CC(C)CC(C)C1)C)NC(c1cc(C(C)C)[nH]n1)=O C1(C)(C(=O)NCCC2N(C(C=NOC)=O)CCCC2)CCCNC1=O C1(NC=O)CN(C(=O)COC(=O)CCC2CCCCO2)C2(CCCCC2)C1.CCF N1(C(C=C(C)Cl)=O)CCN(C(C2CC2C(C)(C)C)=O)C(CCO)C1 C1(CNC(c2nc(COC)sc2)=O)CCCCN(C(=O)C(C)=C(C)CC)C1.CCO C1(CCCNC(C2C(CC)CCC2)=O)CN(C(=O)CN2CCC2)CCO1 C1(CNC(C(CC)O)=O)CC2(CC2)CN1c1nccc(OC)n1 c1(C(C(N2CCC(CC=C)(NC(=O)C=CCSC)C2)=O)C)ccc(OC)c(F)c1 C12(C(=O)NC3CC(CNC(COCc4n(C)ncn4)=O)C3)CC=CCN1CCC2 [N-]=[N+]=NC1CCN(C(=O)CC2CCN(C(c3cc(F)cc(F)c3)=O)C2)C1 N1(C(c2occ(C)c2)=O)CCCCC1C(C)NC(c1cn(C)nc1C)=O CC1CCOC1C(=O)N(CC(O)CNC(=O)CC(=O)N(C)C)C c1(N2C(C)CC(CNC(c3cn(CCO)nn3)=O)C2)ncnc2c1CCO2 N1(C(c2csc(Cl)n2)=O)CC(F)(F)C1C1CCN(C(c2cccnc2)=O)CC1 C#CCC(C)(CC)C(=O)NCCCC(=O)NC1CC2C=CC1C2 N1(C(C2CC(C)(CC)OCC2)=O)CC=CC12CCCC2.C(=O)(C(N=[N+]=[N-])C(C)C)N c1(OC)cccc(CCC(N2CCC3CCC23CNC(=O)C(C)(F)F)=O)c1OC CCC(CC)(CC)NC(=O)CC1CCCC(NC(=O)COCCF)C1 C1(CC)CCCC(C(C(=O)Nc2ccc(C)cc2)N(CC)Cc2cccc(C)n2)C1 C1(OCC(=O)NCC2(F)CC2)CCCC12CN(C(=O)C1CC1)C2 c1(CNC(CN2C(c3onc(C)n3)COCC2)=O)ncc(F)cc1Cl c1(NC(C)=O)cncc(C(N2CC=CC(NC(=O)CC3CCCOC3)C2)=O)c1 c1(COCC(C)C(=O)OC)ccnc(C(=O)N(CCC(=O)NCC)C(C)C)c1 c1(C(N2CCCC(C)(CNC(C(C(C)C)(C)O)=O)C2)=O)ccc2c(c1)CNC2=O n1(CC(=O)NCC(CCOC)NC(C2CNC(=O)C2)=O)nc(C)c([N+](=O)[O-])c1C CCS(=O)(=O)c1ccc(CN2CCCC(C)(C)C2C=Cc2cccs2)cc1 C(C(CC(C)C)C(=O)Nc1ccc(CCO)cc1)NC(C(=O)NC)=O C1(OC)CN(C(=O)COc2ccccc2F)CC1NC(c1ccoc1)=O c1(C(N2CC(CC=C)(NC(c3ccc(F)s3)=O)C2)=O)nccc2cc[nH]c12 CC(C)CCC(O)C(=O)N1CCC(C(=O)NCCCC(C)O)C(C)C1 C1(NC(C2C3CC(NC(C=CC(CC)C)=O)C(C3)C2)=O)CC2C(O)C(O)CC12 CCCC(O)CC(=O)N1CC2CC(C1)C2NC(=O)C(C)OCc1cccc(C)c1 N1(C(CNC(c2c(C)cccc2)=O)=O)CCCCC(CN(C(=O)CC)C)C1.N(C)C C1(C)(C(C2CC2)NC(=O)NC(C2(c3ccc(F)cn3)CC2)C)CC2CCC1C2 c1(CC(=O)NC2C(n3cc(CCCOC)nn3)COC2)nsc2ccccc12 n1(C(C(=O)NCC2(CN(C(CCCC#C)=O)C)CC2)C)c(C)cc(O)cc1=O c1(C(C(=O)N(CCC#N)C2CCC2)NC(=O)OC(C)(C)C)ccc(Cl)cc1 n1(CC(=O)NC(C)CCCNC(C2CC2C2CCC2)=O)cc2ncccc2n1 c1(N2CC(F)CC(NCc3scc(C)n3)C2)ncc2ccccc2n1 c1(-n2cc(CCC(C)O)nn2)n[nH]c2c1CN(C(=O)CC1CSCCO1)C2 Cc1cc(C(=O)NCC(=O)NCC(N2CCC=C(Cl)C2)=O)ncn1 c1(C(=O)NC(CC=C)C(=O)NC(c2cccnc2)CO)cc(F)ccc1F c1(C(N(C2CCN(C(CCC(=C)Cl)=O)CC2)C)=O)ccc(O)cc1F n1(CC(=O)NC2(CC(=O)NCC(F)CO)CCC2)cc(CO)nn1 n1(C(CC)C)nccc1C(=O)NCCCCNC(=O)C(c1ccncc1)C1CC1 C(=O)(CC(C)(C)C#N)NC1CCC(N(C(=O)C(C2(O)CCCCC2)F)C)CC1 Cc1ccn(C(C)C(=O)NCCC(Cc2ccccc2)NC(C2CC(O)C2)=O)n1 Cc1ccc2c(C(N3CC(CCNC(=O)CCC4CCCCO4)C3)=O)n[nH]c2c1 N1(C(CN(C2CCCC2)C)=O)CCC2(CCC2NC(C23CC(CO)(C2)C3)=O)CC1 CC1C(C(=O)NCCCN(C)C2CC2)CCCN1C(c1cncn1C)=O CC#CCC(C(=O)NCCN1CCOCC1)NC(c1cnn(C(C)C)c1)=O c1(C(C(=O)NCC=C)N(C2CCN(CC)C2)C)cccc2c1oc1ccccc21 c1(CNC(c2ccc(C)s2)=O)cc(O)nc(CNC(c2ccc(F)cc2)=O)n1 C1(CC(=O)NCC(CNC(CC2(NC(C)=O)CC2)=O)(C)O)CC(C)(C)CCO1 n1(CCCOC)cc(C2CCN2C(C2CCSCC2)=O)nn1.C12OCCC1NC2=O C1(CNC(C(CC)n2cncn2)=O)CCCCN(C(c2cc(C)c(C)s2)=O)C1 c1(C(=O)OC)ncc[nH]c1=NCC1CC2CCC(C1)N2C(=O)C(C)CC(N)=O CCC(C)CCC(O)CC(=O)N1CC2(NC(c3cncc(CO)c3)=O)CC1C2 C(=O)(CCCC(=O)N1CCC(C(N2CC(OC(=N)O)C2)=O)C1C(C)C)OC S(=O)(=O)(c1ccc(N(CCO)CCO)c(Br)c1)NC(C1(C)CCCCCC1)=O C(CC(=O)N(C1(CO)CC1)C)(C(C)OC)NC(c1nn(CC)c(C)c1)=O c1(C(N2CC(C)C(NC(C#CC(C)C)=O)C(C)C2)=O)nn(C)c2ccccc12 C1(C(C(N2CCNCC2)C)=O)CCCN(c2cnccn2)C1=O C1(C(N2CCC(COC)(CNC(=O)C(=O)N(C)C)C2)=O)CC2(C1)CC(F)(F)C2 C(CCN(C)C(c1cnc(CN)nc1)=O)(C(C)C)NC(c1ccc(COC)[nH]1)=O c1(CNC(=O)NC(c2ccc(C)s2)CC)ccc(-c2nc(C(C)(C)C)cs2)cc1 N1(C(CC(CNC(C(COC)(C)COC)=O)C2CC2)=O)CCC2(CO)CCCC12 c1(NC2(C)CC(NC(c3cc(CO)sc3)=O)C2)cnc2cccnn12.C1(=O)CO1 C1(C#CC(=O)NCC2CC2CNC(=O)CCCCC(C)C)(CC)COC1 C1(OC)CC(CNC(=O)CC(C)(C)c2ccc(C)cc2)N(C(C2CC2CF)=O)C1 c1(OCCC(=O)NCC(C)N(C(C=COCC)=O)CC)cccc(Cl)c1 c1(C(N(C)CC2CCN(C(C(CC=C)CC)=O)C2)=O)cnc2c(c1)NCC2 Cc1[nH]c(C)c(C(N2CC(N(C)C(c3cccc(Br)c3C)=O)C3(CC3)C2)=O)c1C N1(C(CCC=CC)=O)CCC(C(=O)NCCCOCCOC)(CF)C1 N12CCC(CC(N)=O)(CC1)NCC2=O.C(=O)(C(C)C(C)(F)F)NS(C)(=O)=O C(c1ccccc1Cl)=C(C)C(=O)NC(C)(C)C.N12CC(CC1CF)OC2=O C(=O)(CCCC(=O)NC(C1(CNC(C2CC(C)(C)C2)=O)CC1)C)OCC N1(C(C(C(C)C)C)=O)CC(C)(C)OCC1CNC(=O)C1=CCCC1 c1(C(c2n(CCCC)nnn2)NC2CCCSCC2)csc2ccccc12 Cc1c2ccc(NCCCCn3cc(COc4ccccc4)nn3)cc2nn1C c1(NC(c2c(NC(c3c(OC)csc3)=O)cccc2F)=O)n[nH]c2c1CCCC2 N1(C(C(CCOC)NC(=O)CC2C(=O)NN=C2C)=O)CCN(C)CC1C1CC1 N1(C(c2n[nH]c(C)c2Br)=O)CC2CC1CCN2C(=O)CN1CC2CCC1C2 c1(C(N2CC3CC3(C(=O)Nc3nccs3)C2)=O)cc2cc(Cl)cc(Cl)c2[nH]1 N1(C(C(c2ccc(I)cc2)=O)=O)CCC(O)(c2cn(C3CCOCC3)nn2)CC1 N1(C(CCN(CC)CC)=O)CC2CC(CNC(c3cncc(Cl)c3Cl)=O)C2C1 O=C1NC2(CO1)CC(C(=O)NC1CC(CNC(c3cccc4c3CCO4)=O)C1)C2 c1(OC)ccc(C(=O)NC2CCCCCC2NC(=O)Cn2nccc2C)c(F)c1 N1(C(C2CCN(C)CC2)=O)CCC(F)C(NC(=O)Cc2cccs2)C1 C1(CC)CCC(NC(=O)C(=O)NC2CCCC2c2ccncc2)CC1 c1(N2CCCC(NC(C3(C=C)CCOCC3)=O)C2)ncc2ncn(C)c2n1 Cc1cnccc1NC(=O)C(N1CCN(S(=O)(=O)C(C)C)CC1)C C(CCCC(=O)NC(CNC(=O)CSc1n[nH]c(O)n1)C1CCC1)SC C1(Oc2c(Br)cncc2)CN(N2CC(C3CCCCC3)C2)C1 c1(CC(=O)NCC2CN(CC3CC3)CCCO2)c[nH]c2cc(Cl)ccc12 N1(C(c2c(C)nc(C)o2)=O)CCC2(CC2)CC1C(N1CCC(F)(F)C(F)C1)=O N1(C(C2(F)CCC(C)CC2)=O)CCCC2(C1)CN(C(=O)C(C)C#N)C2 C1(CC(=O)NC2(C(=O)NC3CC(OC(C)C)C3(C)C)CC2)CN2CCC1CC2 C1(CNC(c2cc(C(N)=O)oc2)=O)COCCN(C(C2CCCS(=O)(=O)C2)=O)C1 C12(C(N3CCC(NC(CN4CCC(C)CC4)=O)C(O)C3)=O)CCCC1CC(=O)C2 C1(Cn2cc(CCCC(C)=O)nn2)CC12CCN(C(=O)COC1CCCC1)CC2 C(=O)(C(O)CCCNC(C1CC(=O)OC1(C)C)=O)NCCN(CCCF)C C(C#Cc1ccc(C(=O)O)cc1)NC(=O)C=Cc1ccc(F)cc1 C1(F)(CNC(C(C)N(C(C)=O)C)=O)CCN(C(=O)Cc2ccc(Br)cc2)C1 c1(CCCC)nc(C)c(C(=O)NC2(C)CCN(C(c3cnccc3C)=O)C2)s1 N1(C(CC(C(=C)C)O)=O)CCC2(CCCC2NC(=O)C=CCCC)CC1 C=C(C)CC(C(=O)NC1CCNC1=O)NC(=O)CC1CCCN1C C1(NC(c2nnc(C)s2)=O)CN(C(C2CC(C)(F)C2)=O)CC1C1CC1 N1(C(c2n(C)ccc2)=O)CC(CNC(c2cc3scc(Cl)c3[nH]2)=O)CC12CCC2 N1(C(C(c2scc(C)n2)C)=O)CCC2(CC1)CC(O)CNC2=O c1(C(=O)NCCN(C)C(C2OCCO2)=O)cc2nc[nH]c2cc1[N+](=O)[O-] c1(C(N2CCC(N(C)C(c3ccc(=O)n(C)c3)=O)C2)=O)cccn2c(O)nnc12 Cc1ccncc1CC(N1CC(NC(=O)Cc2ccsc2C)C(C(F)F)C1)=O N1(C(c2ccnc(OC)n2)=O)CC2(C)CC1(C(N1CCC(NC(C)=O)C1)=O)C2 CC1(C)C(C(=O)NCC2(CNC(C3CC3(C)C(F)F)=O)CC2(F)F)CC1(F)F C(CCCC(=O)NC1(C2CCCN2C(=O)C=CC(C)(C)C)CC1)SC C(=O)(CCN=c1[nH]ccs1)N1C(CNC(c2cc(C3CC3)[nH]n2)=O)CC(OC)C1 c1(N(CC)Cc2ccccc2F)nccc(=NCc2nocc2C2CC2)[nH]1 n1(C(C)C(C)(C)C)nc(-c2ccn(C)n2)nc1C(c1cccc(F)c1)n1cncn1 C=CCC(CC)C(=O)NCC(C(N1CCCC(C)(C)C1)=O)N(C)C c1(C(N2CCC(C3N(C(CSC)=O)CCCC3)C2)=O)cnn2cccc(Cl)c12 Cc1cc(NC(=O)NCC2CC(C)CN(C(C3CCCO3)=O)C2)ccc1Br CN1CCN(C(c2cccnn2)=O)CC1CNC(C1CCCN1C(N)=O)=O N1(C(C(C(CC)C)O)=O)CCCC(C)(C)C1CNC(=O)CCCCCOC(C)C c1(CN2CCCC(C)(C(N(CCC)C(C)C)=O)C2)cnc2ccnn2c1 N1(C(CNS(NC)(=O)=O)=O)CC(NC(c2ccsc2)=O)CC12CCCC2 C1(C(N2CCN(C(C(CC)c3ccccc3)=O)CC2CC)=O)CC2(C1)CC1(CC1)C2 c1(C(N2CC3C(C(N4C5COCC4C5)=O)C3C2)=O)cc(O)ccc1F N1(C(C2CC(C(=O)OCC)C2)=O)CCCC2(CCC2)C1C N1(C(c2c(CC)nn(C)c2)=O)CCN(C(c2cc(OC)nn2C)=O)C2CCC12 c1(CC)nc(C)c(C(N2CCC(NC(=O)C(C)(F)c3ccon3)C2)=O)o1 n1(CCNC(C2(C(C)C)COC2)=O)cc(C(=O)NC(CO)CCO)nn1 C1(C(=O)NCCC#C)CCC(C)CN1C(C1CC(C)(O)C1)=O CC(CN1CCOCC1)C(=O)N1CCC(CNC(=O)COCCc2cccs2)C1 c1(OCC)cc(C(=O)Nc2c[nH]nc2C(=O)NC2CCCCC2O)cc(O)c1O C1(C)(COC)CC(NC(=O)C(F)(F)CN(C)C)CN1C(=O)CCOC1COC1 C(=O)(C1CCCc2ccnn21)N(CC(=O)NOCC(F)(F)F)C1CC1 c1(OC)ccc(C(N2CC(CF)(NC(C3CCNC(=O)C3)=O)C2)=O)cc1C C(=O)(CCCCCC(C)(C)C)NC(CCNC(C(C)C(F)F)=O)Cc1ccccc1 c1(C(=O)NC2C(C(C)C)N(C(c3cc(C(F)F)[nH]n3)=O)CC2)cn2ccsc2n1 Cc1[nH]cc(C(N2CCCC2CN(C(=O)C(C)(C)F)C)=O)c(=O)c1Br C1(NC(c2c(C)nn(C3CC3)c2)=O)CCC2CCN(C(C3CC3F)=O)C12 Cc1cncc(C(=O)NC2CCC2CNC(c2sccc2C(F)F)=O)n1 c1(C(=O)NCC(C2CCC2)NC(CC(C)C)=O)cccc2nsnc12 CC1CN(C(=O)Cc2ccc3nonc3c2)CC(C)C1NC(n1nnc(=O)[nH]1)=O c1(CCOC)cn(CC(=O)NC(C)CNC(C2(C(=O)OC)CC2)=O)nn1 N1(C(c2c(C)oc(CO)c2)=O)CC2CCC1C1CN(C(=O)CC3CCCC3O)CC21 C(CN=c1[nH]ccnc1F)(C1CCCCC1)N(CCC)C(C12CC=CC(C1)OC2)=O C1(c2ccccc2)(CC(=O)Nc2cn(CC(C)C)nc2)CCCCC1 N1(CCCNC(=O)NC(C(=O)OC)C(C)C)c2ccccc2C(C)C1 c1(OC)c(C(N2CCCC(CNC(C3CCCS3(=O)=O)=O)C2)=O)cnn1C CCCCN=C(NCCc1cn(C)nc1C(F)F)NCC1CCC(C)(C)OC1 C=Cn1nccc1C(=O)NC1C=CCC(C(=O)NC(C2CCCC2)CC)C1 N1(C(Cn2cc(CNC(c3cc(C)sc3N)=O)nn2)=O)CC(C)N(C)C(C)C1 N1(C(CCC#C)=O)CCCN(C(c2cccc(C#C)c2)=O)C(C)C1 N1(C(c2c(COC)cco2)=O)CC(NC(=O)CCC2CCC(=O)N2)CC(F)C1 CCCC#CC(C)(C)NC(=O)CNC1CC(NC(C2(C)CCC(=O)NC2)=O)C1 C(=O)(C(C)(CNC(c1cnc(CC)cn1)=O)CC)N1CC(CCC)C1 C1(C(=O)NCCC(C(C)C)NC(=O)CSC(C)(C)C)CNC(=O)CC1(C)C C1(C)(C(=O)NCCOCCN(C(c2ccc(C)c(C)c2)=O)C)CC(C)OC(C)C1 c1(OC)cc[nH]c(=NCCC2CC(NC(=O)CC3CCCOC3)C2)n1 c1(C(N2CCC(NC(C(CC(=C)C)C)=O)C2)=O)ccc(OC)c2ccncc12 N1(C(CN(C)Cc2ccccc2)=O)CC2CCC1C(CNC(=O)C=CC(C)(C)C)C2 c1(NC(=O)OC)csc(CS(=O)(=O)NCCNC(C)=O)n1 C(=O)(CC(C)CC(C)C)NCCC(C(=O)NCCC(=O)NC)O C12(C(N3CC(COC)(COC)C3)=O)COC(CF)(C1)C2.c12ccnc(c1)C2 c1(CC)cc(C(=O)NC2CCC(NC(=O)C(C)(C)n3cnnn3)CC2)cc(O)n1 CCC(C)(CNC(C1CC=CCN1C(=O)CCCCC1CC1)=O)C(C)O C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C)(NC(CCCC(=O)NCCC)=O)C1 C1(CC(=O)NCC(C(C)(C)C)O)CN(C(=O)C(C)(O)C2CC2)CC12CC2 Cn1[nH]c(=NC(=O)N2CCC(CC3CC3)C2)cc1C(N)=O CC1CCCC(C)CN1C(c1cccc2c1CCC2)C(=O)NCC(F)F c1(OCC)ccccc1OCC12CC(CCO1)C2.C1(c2ccccc2)C(C)(C)N1 C(=O)(N=c1cc[nH]c(C)c1C)C1CCC(CNC(C2C(C)=C2)=O)CC1 C(=O)(CCC(C)(C)C#N)N1CCC(CSC)CC1C C1(CCC)CN(C(=O)C(C)C2(O)CCC2)CC1C(N1CCOC(COC)C1)=O C1(C(N2CC(O)(CNC(CCc3ccc(OC)cc3)=O)C2)=O)CCOC(=O)CC1 c1(CNC(CCN(C(=O)NC)C)=O)cc(C(=O)N(CCCOC)C)no1 CC1(C)OCC(C(=O)NCC2(C)CCN(C(=O)CCSC(F)(F)F)C2)O1 c1(-c2ccc(COC)s2)cn2cc(C(=O)NCc3ccn(C)n3)ccc2n1 C(=O)(C(O)CC(C)C)NC(CC(C)NC(C(C)=C(C)C)=O)C C(=O)(C(C)CC(C)(C)C)N1CC(C(N)=O)(CNC(c2cc(C(=O)OC)[nH]c2)=O)C1 C1(CCC(=O)NC(CN(C(c2sccc2Br)=O)CC)C)CCCN(C)C1 N1(C(c2c(NC)ccc(F)c2)=O)CCC2(CCC2NC(C2(F)CCCC2)=O)CC1 c1(C(N2CC(C(N)=O)(CNC(=O)CC3=CCCC3)C2)=O)cc2c(O)cccc2[nH]1 C1(C)(CC(=O)N(CC(C)C)CCC)CN(C(=O)Cn2cc(C)cn2)C1 S(=O)(=O)(c1cncc(Br)c1)N1C(C(=O)Nc2c(C)ncc(C#N)c2)CC(O)C1 N1(C(c2cc(C)c(O)nn2)=O)CCN(C(=O)Cc2c(Cl)cnn2C)C2CCC12 C1(C(C)C)CN(C(=O)COc2ccccc2)CC1C(=O)NCC(O)CN1CCC1 C(=O)(C(CC(C)C)N(C)C)N1C(CNC(CCc2onc(C)n2)=O)C(C)CC1 C(=O)(CCC(C)(C)F)N1CCCC(CN(C(c2c(C)n(CCO)cc2)=O)C)C1 N1(C(c2cn(CC(=O)OC)nc2)=O)CC(NC(c2ccc(O)cc2)=O)C(C)C1 c1(NC(c2ccc(SC)c(C)c2)c2n(CCOC)nnn2)ccc2c(c1)COC2 c1(NC(=O)NC(C(c2cccnc2)OC)C)ccc2c(ccn2CC(C)C)c1 CCC(CC(C)CO)c1nc(-c2ccnc(OC)c2)nn1C1CCC(OC)CC1 c1(C(N2CC(CCC)N(C(=O)Cc3cncs3)CC2)=O)cnc2sccc2c1 C#CCC(C)(C)C(=O)NCC1CN(C(=O)C2=CCCC2)CCCO1 C1(C2CCCO2)(C(=O)NCC(CNC(c2c(C)snc2)=O)(C)O)CCOCC1 Cc1cc(C(N2CC(C3(Nc4nnc(C)c(C)n4)CC3)C2)=O)cc(F)c1 CCCCCC(O)C(=O)NC(C(=O)NC1(C(N)=O)CC1)C1CCC1 C(=O)(CCCC(=O)NC(C)C)N1CCC(CNC(CC(CC)C2CC2)=O)CC1 N1(C(c2ccc3ccoc3c2)=O)CCC2CCC(C1)N2C(c1snc(O)c1Cl)=O CCC(C)CC(=O)NC(Cn1cncn1)C(=O)N(C)CC1(F)CCC1 Cc1nc(NCCCOCCCO)cc(NCCCC2CC2)n1 N1(C(C2C(c3n(C)cnc3)C2)=O)CCC2(NC(=O)CC3CC3(Cl)Cl)CCCC12 N1(c2nccc(SC)n2)CCC2(CC(NC(c3cc(-c4ccco4)on3)=O)C2)C1 N1(C(CCC(=C)C)=O)CC(C)CCC1CNC(c1ccn(C(C)C)c(=O)c1)=O N1(C(c2c(C)n(C(C)C)nc2)=O)CCCN(C(=O)C(C)Oc2ccccc2)CC1 c1(C(N(CC(CC)NC(=O)C(O)CN2CCCC2)C)=O)cccc2nonc12 C(CCN=C(NCCc1ccc(Cl)nc1)NCC1CCC(C)O1)NC(COC)=O N(C(=NC(C)C)N1CCC(O)C1)CC(CC)Oc1ccccc1 C1(CCC)(C(N2CC(O)CC2CNC(=O)COCC(F)F)=O)CCNC1=O C1(O)(CN(C(C(=O)NCCOC)=O)C)CN(C(C2C=CC2C(N)=O)=O)C1 C(c1c(Cl)cccc1Cl)=C(C)C(N1CCC(F)(CNC(C2(C)CCCS2)=O)C1)=O N1(C(c2ccn(C)c2)=O)CCC2CN(C(c3cc(C4CC4)ns3)=O)CC2CC1 N1(CC(N2CC(OCCNC(C(C)NC(CC)=O)=O)C2)=O)CCC(C)CC1 c1(C(=O)OCC)c(-c2ccc(C(C)CC)cc2)cnn1C C(=O)(C(CNC(c1n[nH]c2c1COC2)=O)C(C)(C)C)NC(CC)(CC)CC Cc1cccc(F)c1CC(=O)N(CC(O)CN(C)C(c1cc(Br)cn1C)=O)C c1(NC(c2nccc(C#C)c2)=O)nc2c(s1)CC(NC(=O)C(O)C(C)C)CC2 N1(c2c(C)cncn2)CCC(F)(F)C(C(N2CC(O)CC2CN2CCCC2)=O)C1 c1(NC(c2c(CNC(c3ncc(CC)cn3)=O)ccs2)=O)ccc(Cl)cc1C c1(CNC(CC(C(C)C)OCC)=O)nc2c(s1)CN(C(=O)C(O)CC)CC2 N1(C(C2CCC(C)C2)=O)CCc2c(c(CNC(=O)CC3CCCN3C)nn2C)C1 c1(CN=C(NC(C=C)C)NC2CC3(CC3)C2)cccc([N+](=O)[O-])c1C Cc1cccn2c(C(=O)NC3(C4CCN(C(=O)CCOC(C)C)C4)CC3)cnc12 CC(C)CC(O)C(=O)NC1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C12CC2 c1(C(N)=O)cc(C(=O)NC2CC2CNC(=O)CCCOc2cccnc2)co1 N1(C(c2cn(C)[nH]c2=N)=O)CCC(CNC(c2ccc(CO)cn2)=O)C12CCC2 C1(NC(CCOCCOCC)=O)CC2CC2N1C(C1(COCC)CC1)=O N1(C(CC2CC(=O)NCC2)=O)CC2(CCC(NC(=O)CCc3ncc[nH]3)CC2)C1 c1(OC)ccc2cnc(N(c3ncnn4cccc34)C3CCNCC3F)nc2c1 C1(OCC)CCCN(c2nnc(C3CCOC3)n2Cc2csc(CC)n2)C1 C(=O)(C1=CC(C)(C)C1)N1CC(NC(C2C(C(=O)OC)CCO2)=O)C(C)C1 C1(N(C)C)(C(=O)NC2CCC(NC(c3cc(C4CCC4)[nH]n3)=O)C2)CCCSC1 N1(C2c3nccc(c3)NC2=O)CCCC(CO)CC1.C1(C(=O)OC)CC1 Cc1ccn(C(C)C(=O)N(C(c2ccccc2)CNC(C2(C)CC2)=O)C)n1 C1(CN2CC(CC(C)OC)C2)CCC2(CCC2)C1.C1(=O)C(CC2CCOCC2)N1 C1(C(C)(O)CNCc2ccncc2F)CCN(C(=O)OC(C)(C)C)CC1 C#Cc1ccc(C(=O)NCCCCC(CO)NC(=O)C(COC)OC)nc1 C1(C(C)C)CN(C(c2ccnc(Br)c2Cl)=O)CCN1Cc1ccc(O)nc1 C(C(C)C(C)(C)C)OCC.c12cc(ncn1)C(=O)NC1CC(C1)CNC(=O)N2CC C(=O)(CCS(C)(=O)=O)NCC(C(C)C)(C)NC(=O)CCCOc1cccc(F)c1 C(CC#CC)(C(=O)N1CC(O)(CC)C1)NC(c1c(CC=C)cccc1)=O C(=O)(C1=NOC2CCCCC12)N1C2CCC(CN(C(=O)C#CC3CC3)C3CC3)(C2)C1 c1(C(=O)NCCNC(C(c2cscn2)N(C)C)=O)nn(C)c2c1CCCC2 c1(CC(=O)NC(CNC(C2CCSC2)=O)CO)cc(Cl)cc2c1OCC2 C#Cc1cn(C)nc1C(=O)NC1CCC(C)(CNC(c2ccnc(Cl)c2O)=O)C1 C1(C(=O)NCCN(C(c2cc(C)c(C)o2)=O)C(C)C)CC2(CCCCC2)S1(=O)=O C(=O)(C(O)CCCNC(=O)CC1CC(OC(C)=O)C1)NC(C1CCCCC1)C#C C1(CNC(c2c(C)cc(SC)o2)=O)CCCCCN1C(=O)Cc1cncc(O)c1 C1(C(=O)NC2CC(C#N)(OC)C2)CCN(C(=O)CCCC2CCC2)C(C)C1 c1(NC(c2c(NCc3c(C)cccc3F)cnc(Cl)c2)=O)cccn2cncc12 CCS(=O)CC(=O)NCCCC1CCN(C(c2ccnn2COC)=O)CC1 CN1CCC(C(N2CC(NC(c3cc(C(F)F)n(C)n3)=O)C(O)C2)=O)CC1 Cc1ccsc1CNC(C1CCCN1C(=O)NC1(c2ccccc2)CC1)=O c1(NC(CC)(CNC(c2c[nH]cc(Cl)c2=O)=O)CC)c(C)cccc1[N+](=O)[O-] n1(CCOCC=C)c(N2CCC(NC(C)=O)C2)nnc1-c1sc(C2CC2)nc1C C1(N(C(=O)C(O)C(F)F)C)CC2CCC(C1)N2C(c1ccc[nH]1)=O N1(c2cc(N3CCC(C(N)=O)CC3)nc(C(F)(F)F)n2)CCn2cnnc2C1 C1(CNC(C(F)=CC)=O)C(C)CCCN1C(c1ccn(C(C)C)c(=O)c1)=O c1(C(N2CC3C(CNC(=O)Cc4cnoc4)(C3)C2)=O)coc2c1C(=O)NCCC2 C(C(C)CC(=O)N(C1CCC1)C)NC(c1nc(CC)oc1)=O c1(CCCC)ncc(C(=O)Nc2ccc(=O)n(Cc3ccccc3)c2)c(C)n1 CN1CCN(C(C2CCCCNC2=O)=O)CC1C(=O)N(C1CCN(C2CC2)C1)C CC1(C)CCC(CC(=O)OCC(N2CCN(CCOc3ccc(Cl)cc3)CC2)=O)O1 c1(OC)c(C(N2CC(NC(C3CCCO3)=O)CC3(CC3)C2)=O)cccc1[N+](=O)[O-] C1(N(C(CSCC(=O)OC)=O)C)CN(C(=O)CN2CCC(C)(C)C2)CC1(C)C c1(C2(NC(c3n(SC)nnn3)CCC3CCCOC3)CC2)ccc(C)c(F)c1F C(=O)(CCCC(=O)NC1CN(C(C2CC(O)CN2C(N)=O)=O)CC1O)NCC CCC(CCC(=O)NC1CCCC1)N(C)C(C1CCOCC1)=O c1(C(N2CC(NC(CCCOC(C)C)=O)C(F)CC2)=O)cc2n(n1)CCCN2 C=CCCC(C)(C)C(=O)N(C(C)C(=O)NCC1(CO)CCOC1)C1CC1 C1(N2CCCC(NC(C(N3CCC(C)(F)CC3)C)=O)C2)CCC2(CCC2)CC1 C(=O)(C1=NNC(C(F)(F)F)C1)NC(C1CN(C(C2(O)CCSCC2)=O)C1)C C12(C(=O)NC(C)C(=O)NC(C)(C)C)CC(NC(c3ccnnc3)=O)(C1)C2 C1(N(c2ccc(C)c(O)c2)C(c2ccc(O)nn2)=O)CCCC12CCNCC2 C1(CC(=O)NCCN(C(CCC(=O)NC)=O)CC2CC2)CC2C=CC1CC2 C#CC(CO)(CO)NC(=O)C(C1CN(C(=O)CC2COCC(C)O2)C1)OC c1(C(=O)NCc2c(C(N3CC(C)SCC3)=O)occ2)cc2ccccn2c1 N1(C(CC2(C(=O)OC)CC2)=O)CCC2(NC(c3cc(C)ccc3F)=O)CC2C1 CC1CCCN(Cc2ccc(-c3ccc(Cl)cc3)c(F)c2)C1C N1(C(C(=O)NCC)=O)CCc2c(COC)cccc2C1.C1CCCCCO1 CC1(C)CC(O)(CC(N2CCC(NC(=O)CN3CC(C)(C)C3)CC2)=O)CO1 CC1(C)CCN(C(C2CC(=O)C23CCCC3)=O)C(C(N2CCS(=O)CCC2)=O)C1 N1(C(C(CC(C)C)OC)=O)CCC(NC(=O)CCC(C)(C)O)C12CCC2 c1(CNC(c2ccco2)CC)c(C)nn(C(F)(F)F)c1C Cc1nnc2n1CCCC2C(=O)NCCCNC(C1CC(C2CC2)=NO1)=O N1(C(C=CCC(C)(C)NC(CC(CC)C2CC2)=O)=O)CCC2CN(C)CC2C1 C1(CNC(=O)CCC2CCCCO2)(NC(c2ccncc2F)=O)CCCCC1 C1(C(=O)NCC(C)N(C(c2c(C)snc2)=O)C)CC(=O)N(C)C1c1cccnc1 C1(CC)CCN(N2CCC(CNC(=O)OC(C)(C)C)CC2)CCO1 N1(C(C2(C(F)F)CC(=C)C2)=O)CC(NC(=O)Cn2nc(C)c(Cl)c2C)CC(C)(C)C1 C1(CNC(c2scc(C(C)=O)c2)=O)(N)CCCCC1.N1(C(=O)C(N)=O)CCCC1C c1(C(N2CCCC(C)(O)C2)=O)cc(O)nc2c1CN(C(C1C=CCS1)=O)CC2 O=C1NC(=O)C(CC(N2CC3CC2C3CNC(=O)C(F)n2cccn2)=O)N1 CC1(N)CCCCC1NCCCc1cccc(C(N)=O)c1 N1(C(=O)NC2CC(C(=O)OC)OCC2)CC=CCC12CCCCC2 N1(C(C2(C)CCCN2C(c2cnc(N)cn2)=O)=O)CCc2ccncc21 c1(C2(O)CCN(CC(=O)N(c3ccccc3)CC)C2)ccc2n[nH]cc2c1 C(=O)(C(C)CC(F)(F)F)N1CCC(C(N(C2CC3CC3C2)CC)=O)(CF)C1 C1(C(=O)OC)CC(c2cn(C3CCOC3)nn2)CN1C(C)C(=O)OC CC1CCN(C(=O)Cc2cc(C3CC3)no2)CC1N(C(=O)CCc1nccs1)C C(=O)(C(C)P(C)(C)=O)NCc1ccc(CC(C)NC(=O)Cc2cncs2)cc1 C1(COc2cc(C)c(NC(c3cccnc3)=O)cc2)CCC2(CCNCC2)O1 c1(C(=O)Nc2cnn(C3CCOCC3)c2)ccc2nc(Br)nn2c1 C(=O)(C(CO)C(C)(C)C)NCCC(CCNC(c1nc(C)oc1)=O)C C1(NC(C(=O)NC(C)CS(C)(=O)=O)=O)CCCCC(P(C)(C)=O)C1 c1(CCC(=O)NC(C(C)NC(c2ccc(C(C)=O)o2)=O)C)nnc(S)nc1O N12CC3(CO)CC1(C3)C2=O.C1(OC)CCC(C(=O)NC2CC(n3cncn3)C2)C1 C=C=C(C)CC(=O)NC(C)C(C(C)C)NC(c1ccnc(C)c1)=O Cc1cc(F)cnc1C(=O)NC1(C)CN(C(=O)CN2CCCCC2C)C1 c1(C(N2CCCC(C)(CNC(C3(C(F)F)CCC3)=O)C2)=O)cc(Cl)c(O)c(Cl)c1 N1(C(c2ccc(SC)s2)=O)C2CCC1CN(C(c1cnc(C3CC3)o1)=O)CC2 C1(NC(C(C)CF)=O)CCC(CN(C)C(c2cccc(Cl)c2)=O)CC1 Cc1ccc(COC(C)CN(C(=O)CCN(C)C(C2CC2C)=O)C)cc1 C(CC)(CC(=O)NCc1cnc(C)n1CC)NC(CC#C)=O c1(C(N2CCN(C(CC3CC(=C)C3)=O)CC2CC)=O)ncn2ccccc12 C1(CC#C)(C(N2CCCC2c2cn(C3CCOC(C)C3)nn2)=O)CCCCC1 c12cc(C(=O)O)c([nH]1)C2.c1(CC(C)C)cn(C2CN(C(C3CCC3)=O)C2)nn1 N1(C(c2c(OCC)ccs2)=O)CC(NC(c2cc3n(n2)CCC3)=O)CC(O)C1 c1(OC)ccc(F)c(NC2CC(C)N(C(=O)OC(C)(C)C)C2)c1 C1(C(=O)NCCCN(C(c2c(Cl)cnc(O)c2Cl)=O)CC)CN2CCCN1CC2 C1(C)(CN(C(c2cc(C)on2)=O)C)CCCC1NC(=O)C=CSc1nc[nH]n1 C1(C(C)C)CN(C(=O)OC(C)(C)C)CCCN1C(c1cccc(CCF)c1)=O C1(C(N(C2CCCN(C(=O)C=C3CCC3)C2)CC2CC2)=O)CC2(CCC2O)C1 C1(CNC(C2CC2F)=O)COC(C(F)(F)F)CN1C(=O)C=Cc1ccco1 c1(C(=O)NC2CC(n3cc(C(C(C)C)(C)C)nn3)C2)ccc(C#N)c(Cl)c1 O=C(C1=COCCC1)NC1(CNC(=O)CC2CCC2)CC2CCC1C2 C(=O)(C(C#N)C(C)C)N1C(=C(C)C)C(NC(=O)C=CCN(C)CC)CC1 c1(CCC(N2CCCCC(NC(C(F)=CC)=O)C2)=O)csc2ccccc12 N1(CCC(=O)NCCC(CNC(=O)CC2CS(=O)(=O)C2)CO)CCCCCC1 c1(CC(=O)OC(C)(C)C)cccc(N(C2CCCC2C#N)C(OCOC)=O)c1 N1(C(C2CCC(C)O2)=O)CC2CCC1CN2C(=O)C=CC(=O)N(C)C1CC1 N1(CC(=O)N(CC(CC)NC(C(C=C=C)C)=O)CC)C(=O)c2cccnc2C1=O N1(C(c2ccc(C)s2)=O)CC(n2cc(CO)nn2)C(C)C1.c12cccc(c1)CO2 C1(CNC(CC2C(C)C2)=O)CCCN1Cc1nc(C2CC2)n[nH]1 CCCCCC(C)CC(=O)N1CCC2CN(C(=O)C(C(C)C)OC)C(C)C12 c1(-c2nccc(C(=O)NCc3c(OC)n(C)nc3)c2)ccc(SC)cc1F Cc1cnn2c1CN(C(=O)C(CC(C)(C)C)NC(=O)CSC(F)F)CC2 C1(NC(c2c(C)ncc(Cl)c2)=O)COC2(C1)CN(C(=O)Cn1nnc(=N)[nH]1)C2 Cn1cc2ccc(C(=O)NC3COCC3NC(C3CSCCS3)=O)cc2n1 C(=O)(C(CN(C)C)CC)NC(C(=O)N(C(CCC)C)C1CC1)C N1(C(C(CC)N(C)C)=O)CCC(NC(c2cnc3[nH]cncc2-3)=O)C(C)(C)C1 C12(CNC(C3N(C)CCC3)=O)CCCCC1N(c1ccc(S(C)(=O)=O)cn1)CC2 N1(C(C(CCCNC(=O)CCC2CC2)O)=O)CCC(O)(C2CC2)CC1 C#Cc1cn(C)nc1C(=O)NC(c1ccc(F)c(Cl)c1)CO C1(C(=O)NCC2C3CN(C(c4n(CCC)ncc4)=O)CC32)CCCCC12CCC2 C#CCC(C)C(=O)NCC1CCCN(CC2CCC2)C1 N1(C(c2cc3cscc3s2)=O)CCCC(C2CN(c3ncc(Br)cn3)C2)C1 c1(C(=O)OC)cccc(COC(=O)C(C2CCOC2)OC)c1 CCC(O)C(C)C(=O)NCC1(C(C)(C)C)CCN(C(=O)CC#N)C1 N1(C(c2nc(CC)sc2)=O)CCCCC1CNC(c1nccs1)=O Cn1c([N+](=O)[O-])cnc1C(N1CCN(C(=O)CN2CCCC2)CC1)=O C(CC(C)C(=O)NCC(CCOC)NC(=O)CC1(C)CCCC1)OC C1(C(=O)NC2(CCC(=O)NC(C)C(C)n3cccn3)CCC2)CC=CCC1 C(CN=c1[nH]c2c(c(=NCCF)[nH]1)SCC2)N1C(CC)CCC1 c1(C(N2CC(C(C)NC(c3nccnc3N)=O)C2)=O)ccc(F)cc1Cl C(C)(CCI)(C1CCOCC1)NCC(C1CCCO1)OC c1(C(=O)NCC(CC(C)C)NC(=O)C(C)C(F)(F)F)ccc(C(C)C)nc1O N1(C(C(C)S(N)(=O)=O)=O)C2CCC1CN(c1ncnc3c1ncn3C)CC2 C(C#Cc1ccc2cc(C#N)ccc2c1)N1C=C(CC(C)(C)CO)CN=N1 C1(C(C)(C)C)CCCN1C(c1cnn(Cc2nc[nH]n2)c1)=O CC1(C)COC(C(=O)NC2CC(C)(NC(=O)CCOCC(F)(F)F)C2)C1 c1(CCC)cc(C(=O)NCc2cc(C(=O)NCC(C)C(C)O)on2)n[nH]1 C(CC(F)F)(C(=O)N)N(C(c1c(SC)scn1)=O)C.C1(CO)(CO)CCN(C)C1 N1(C(Cc2cn(CC)nn2)=O)CCCCC1CCCNC(C1(C)CNC(=O)C1)=O C1(C(=O)NCC2(Cn3cc(C4CCC(CO)CC4)nn3)CC2)CCC(C2CC2)C1 Cn1cnc(C=CC(N2CCCC(CNC(C3CC3Br)=O)C2)=O)c1 c1(CCN2CCCC(C(N3CC(CN)C3)=O)CC2)cn2c(n1)CCCC2 CN1CCCCC1CC(N1CCC(C)(CNC(=O)Cc2ccoc2)C1)=O N1(C(C2(CCC=C)CC2)=O)Cc2ccccc2C(NC(c2cnoc2)=O)C1 N1(C(CCc2cccc(C)c2)=O)CC2CCC1C2NC(=O)CC1CCCS1(=O)=O c1(C(CCC)=O)csc(NC(=O)OC(C)(C)C)n1.C(=O)(C)NCCNC(C1CC1)=O c1(OC)ccc(Cl)c(C)c1C(=O)NCC1(CNC(=O)CC2CCCO2)CCCC1 CC1CN(C(=O)C#CC2CC2)CC1(C)CNC(c1ccc(-n2cccn2)nc1)=O C1(NC=O)C2CC3C(C2=O)C13.C(CCO)N(C(=O)CC1CCC1)C CCCC(CNC(=O)CC(C)SC)C(=O)NC1CCCCC1CC CCC(C)(C#N)C(=O)N(CCCNC(=O)CCN1CCCCC1=O)C1CC1 CC1(C)CN(CCC(=O)NCCCCNC(=O)CC2CC2(C)C)CCS1 C(=O)(C1Cc2ccccc21)NC(CC)CC(=O)N1CCC=C(Cl)C1 C1(NC(CN(C)CCO)=O)CC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 C1(=CC(=O)NC(CNC(C2(OC)CCCCC2)=O)C2CCC2)CCCCC1(C)C c1(C(=O)NC(CC=C)CNC(C2CC(=O)N2)=O)ccc2c(c1)SCC(=O)N2 c1(CS(N2CC(CCC)OCC2)(=O)=O)ccc(F)cc1F C1(CNC(c2c(SC)scc2)=O)CCN(C(=O)C(C)n2cncn2)CC1C C(C1CCC(C)CC1)=CC(=O)NC(C)C(C)NC(c1cc(Br)c(C#N)s1)=O C(=O)(C(C)(C)C(C)NC(c1cc(F)n(C)n1)=O)N(C)Cc1c(C)cccc1 N1(CC(C)NC(=O)C=CC2CCC2)CCN(C(=O)CCC2CCC(C)O2)CC1 N1(C(C(=O)NC(c2cc(OC)c(F)cc2)C)=O)CCC(OC)C(C)(C)C1 CC(C1CCCCC1)=CC(N1CCN(C(c2ncc(N)nc2C)=O)CC1CO)=O N1(C(C2(C(C)(F)F)CC2)=O)CC2CC(NC(=O)Cc3cnccn3)C2C1 C1(O)(CNC(C2C=CCN(C(CN(C)CC)=O)C2)=O)CCC(C)(C)C1 NS(=O)(=O)c1ccc(C(N2CC3(CCCC3NC(c3cnc[nH]3)=O)C2)=O)c(Cl)c1 N#Cc1ccccc1C(N1CCCOC(CNC(=O)C(Cl)=CCl)C1)=O C12(NC(c3c(CC)n(C)nc3)=O)CCCN(C(c3cc4c(s3)CCC4)=O)CC1C2 c1(C(N(C(C)CNC(=O)C(C)(C)F)CC)=O)nc(C(C)C)ncc1Cl CC1=C(C(=O)N2CC3C(CC(=O)N(C(C)CC(C)C)C)C3C2)CCCO1 CC(C)P(=O)(CC(=O)N1CCC(O)(CNC(c2coc3c2COC3)=O)C1)C(C)C C1(C(=O)NC(C(N2CC(C)(C(N)=O)C2)=O)(C)C)CCCCC1F C1(NC(c2c(C)csc2)=O)CN(C(c2c(Br)noc2C)=O)CC1F C1(F)(C(=O)Nc2c(CC)nsc2)CCCN(C(c2cnc(C)o2)=O)C1 N1(C(C2C(C)(NC(=O)CCCCC3CC3)CCCC2)=O)C2CCC1CC(O)C2 N1(C(C(C(C)C)CNC(C2C=CC=CC=C2)=O)=O)Cc2cnn(C)c2C1 Cc1cc(C(=O)NC2CC(N(C)C(c3cccnc3S)=O)C2)c(N)cc1F C=CCCCC(=O)N1CCCC(C(C)(O)CNC(=O)C=C2CCCC2)C1 C1(CNC(CC2(C)OCCO2)=O)CN(C(C2(P(C)(C)=O)CC2)=O)CC1(C)C C1(O)(CNC(CC2CC(=C)C2)=O)CCCN(C(=O)C(C)C(C)(F)F)C1 N1(Cc2cn(C(C)(C)C(=O)NC3CC3)nn2)CCc2ccc(O)cc2C1 N1(C(c2c(C)cncc2)=O)CCCC12CCN(C(C1(C)CS(=O)(=O)C1)=O)C2 C(CC(C)C(=O)NCc1ccc(C(=O)NC(C)CC(C)C)nc1)OC C1(NC(C2(NC(N)=O)CC2)=O)CCC2CN(C(=O)C3=CCCCO3)CC2C1 N1(C(C2C(C)CC(=O)N2)=O)CCCC2(C1)CN(C(c1cc(N(C)C)ccn1)=O)C2 Cc1c(C(=O)NCC2CC(C)N(C(=O)CC3CC(=O)C3)C2)sc2ccccc12 c1(C(N2CCC(C(=O)Nc3scc(C(C)=O)n3)C2)=O)c(C)nn2cc[nH]c(=O)c12 C#Cc1cn(C)nc1C(=O)NC1C=CC(CNC(=O)C(N2CCC(O)CC2)C)C1 C#Cc1cccc(CC(=O)NCC2CCC(C)CN2C(=O)C(C)C2CCCC2)c1 CN1CC2C(C(=O)N(C(C)(C(=O)N3CCC3C3CCCC3)C3CCC3)CCO)C2C1 c1(OC)cccc(C)c1C(N1CC2(CC(NCc3ccc(Br)c(F)c3)C2)C1)=O c1(CNC2(c3c(C)cccc3)CC2)cccc(C#N)c1.C12CNC(C1)C(=O)NC2 c1(C(N2CC3C(NC(C4CC(=O)NC(=O)N4)=O)C3C2)=O)ccc2nccn2c1 c1(CNC(N2C(CC(=O)OC)C3CCC2C3)=O)ccc2oc(=N)[nH]c2c1 C1(C)(SCC)C=C(C(=O)N2CCCCC2c2cn(-c3ccc(Cl)c(C)c3)nn2)C1 c1(C(=O)NCC2CN(C(COC)=O)C(C)C2)ccn2nnnc2c1 O=C1NCCc2ccc(NC(c3sccc3Nc3nc4ccc(Cl)cc4[nH]3)=O)cc21 C12(CNC(=O)Cc3ccsn3)CCCC1N(C(=O)CCC(F)F)CC2 C(=O)(C#CC1(C)CCCO1)N1CCCC(CNC(C(C(C)C)NC=O)=O)(CO)C1 c1(C(=O)NCCN(C(C(C)NC(C)=O)=O)CC2CC2)cc2n(n1)CC(F)C2 N1(C(C(c2cccc(OC)c2)F)=O)CC(NC(=O)C(C)C)CC(C)(C)C1 c1(-c2nnc(C)o2)ccc(C2CC2)cc1.C12CCCN(C1)c1nc(no1)C(=O)N2 C(CCC(C(=O)NCCCn1cc(Br)cn1)N(C1CC1)CC)OCC C12CCCN1C(=S)NCC2.c1(NCC#C)ccccc1 C1(C(=O)NCC)C=CCN(C(=O)NC23CCC(OC)C2C3)C1 CS(=O)c1nc(CNc2ccc(Nc3ccc(Cl)cc3F)c(Cl)c2)c(N)c(N)n1 C1(O)(C(C)NC(=O)COCC2CCOC2)CN(C(c2ncnn2C)=O)C1 N(C1CCCn2ncnc21)C(C(CC1CCC1)NC(C1N(CC)CCC1)=O)=O CCCCC(CC)C(=O)NCC1CC2CC2N1C(C1CCCCN1C)=O Cc1cc(C(N2CC(C)(NC(=O)CC(O)C3CCCC3)C2)=O)ns1 C1(CNC(c2ccn(C(F)(F)F)n2)=O)(NC(C2CC3(CSC3)C2)=O)CCCCC1 C1(C(=O)NCC(C)(O)CNC(C2CCN(C(N)=O)C2)=O)(CF)CCC(F)(F)CC1 C1(C(N2C(CC)CCC2)=O)CC(F)CCN1C(c1cnn(C)c(=O)c1)=O c1(OCCC)cccnc1NC(=O)CN(C(=O)CSc1cn[nH]c1)C.C1CN1 C(c1cc(F)cc(F)c1)=CC(=O)NC(CC1CN(C(C(CSC)(C)C)=O)C1)C c1(C(=O)NCC(CCNC(c2cccc(CC)n2)=O)OC)cccn(C)c1=O c1(CS)ccc(CO)c(CO)c1.c1(C(C)OCC)ccc(CC)o1 Nc1ccc(C(=O)NC2CC(NC(c3ccccc3F)=O)C23CCC3)c(O)c1 C1(C(=O)Nc2c(CC)nn(C)c2)CC(C)CN(C(=O)CSCC(F)F)C1 c1(CC(C)(C)O)ccc(NC(=O)Cc2csc(Cl)c2)cc1 N1(C(c2nc(C)sc2)=O)CC(C)OC2(CCN(C(c3ccc(C#N)s3)=O)CC2)C1 C(=O)(C(C)(C)C(C)(F)F)NCCCN(C(C1CCC(C(=O)OC)CC1)=O)C(C)C C12COCCC1NCC(=O)N1CC(O)(C1)C(F)C(=O)N2.c1(N)ccccn1.C=CC C(C(C)CC(=O)OC)N(C1CC1O)C(C1CCN(CCF)C1)=O Cc1nc(NC2(CNC(C3(C=C)CC3)=O)CCOCC2)cc(C#N)n1 C1(C2CC2)(C(N(CCCC#C)C)=O)CN(C(c2ccn(CCC)n2)=O)C1 CC(C)(C)CCC(F)C(=O)N1CC2CCC1CC2NC(c1ccc[nH]1)=O C(=O)(C(C)(C)C(C)(C)C)NCC(C(=O)N(C)CC1OCCC1(C)C)N(C)C N1(C(c2cc(C)nn2C)=O)CC(CNC(C2(CO)CC(=O)C2)=O)OC(C)(C)C1 C1(NC(=O)C=CCN2CCCC2)CCCCN(C(=O)CC=Cc2ccccc2)CC1 C1(C(=O)N(C(c2cn(C3CC(C(=O)O)C3)nn2)(C)C)C)(OC)CCOC1 c1(OC)nc(=NC(C)c2nc(O)n[nH]2)[nH]cc1Br Cc1cc(C(=O)NCC2(CCNC(=O)C3=CCCC3)CC2)nn1C(=O)NCCN C1(NC(c2c(C)cco2)=O)CC2CCC1CC2NC(=O)CC1CCS(=O)(=O)C1 CCCCC(CNC(C1(C(=O)NC)CC1)=O)NC(=O)C(Cc1ccccc1C)CC CC1CCC1C(=O)N(C1(CC(=O)N(C)CC2CC2(F)F)CC1)C N1(C(C)=O)CCCc2cc(CNC(=NCC3(C)CCOC3)NC(C)C)ccc21 n1(CC(NNC(=O)C(C)C)=O)cc2c(n1)C(NCCCCCCCCBr)CCC2 C12(CNC(Cn3c(CCC)nnc3S)=O)CCC(CC1)N2C(c1cc(C)no1)=O CC1CN(C(=O)OC(C)(C)C)CCC1C(=O)Nc1ccc(SCC#N)cc1 C(=O)(C1=CCCS1)NC(c1ccccc1)C(C)NC(C1(CCC=C)CC1)=O CC1CCC=C1C(=O)N1CCN(C(=O)CN2CCCCC2=O)CC1c1cn[nH]c1 C1(C(=O)NC2CC(NC(=O)C=Cc3ccccc3F)C2)CC2(CCOCC2)C1 C12(CNC(C(N)=O)=O)CCCC1N(C(c1ccc(Br)c(O)n1)=O)CCC2 c1(CN(C(=O)C(=O)NC2CC2)C)cc(F)cc(N)c1N.C12CCCN1C2 c1(C(=O)NCC2C(NC(C(=Cc3cnc[nH]3)C)=O)C2)cc2ccncc2[nH]1 c1(-c2cn(C3CCC(C(N(CCOC)C(C)C)=O)C3)nn2)c(C)cccc1Br c1(C(=O)NCCCC(C)NC(CC=C)=O)ccc(OC)c(OC)c1Cl N1(C(c2c(C)c[nH]n2)=O)CCC2(CC1)CC2NC(C1CCC(N(C)C)CC1)=O C1(NC(c2c(C)snc2)=O)CCN(C(=O)CC2CCCC23CC3)CC(C)(C)C1 N1(C(Cc2c(C)cco2)=O)CCCC(N(C(=O)CCOC(C)C)C)C1 C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1CCC(NC(c2c(CC)[nH]nc2Cl)=O)C1 c1(NC(C(C(CC)C)NC(=O)OC(C)(C)C)=O)nc2ccccc2s1 c1(NC(C2CCN2Cc2ccc(Br)nc2Br)=O)cnc2cc[nH]c2c1 Cc1[nH]c2ccccc2c1CCNC(=O)COC1CN(C(c2cncnc2)=O)C1 CC(C)(CNC(C1CCSCC1)=O)CC(=O)NCC1C=CCC1 Cc1noc(C)c1.N1(C(C2(C3NC(=O)NC3=O)CC2)=O)CCC(NC(=O)C)C1C Cc1nc[nH]c1CC(N1CCCC1CNC(=O)Cc1ccnn1C)=O C(C(C)(C)C(=O)NCc1cnn(C)c1C(N1CCCC1(C)C(C)O)=O)OC(C)C N1(C(C23CCC(C)(C2)CO3)=O)C2CCC1CC(NC(=O)CC1COCCO1)C2 C(=O)(C1c2c[nH]nc2CCC1C)NC1CN(C(C(C)=C(C)C)=O)C1 C(=O)(C1CCCc2c1ncn2C)N(C)CC1CC(C(=O)OC)C1(C)C C(=O)(C1CCCc2ccccc21)NCCNC(=O)C=CCl.C(CC(=O)NC1CC1)N C12CC3CC(C1)N(C3)C(=O)CCc1cn2nn1.C(CCCCCO)OC N1(C(C(C2CC2)SC)=O)CC=CC(C(=O)NC)C1.C12(CCSCC1)C(=O)N2 C(=O)(C1CCCn2cnnc21)N1CC2(N(C(CCc3c(C)noc3)=O)CC2)C1 CCC(CC)(CC)C(=O)NCC(C1CCCN1C(c1nc(Cl)c(Cl)s1)=O)(C)C N1(C(C2CC(C)(CC)OCC2)=O)CCC(C)C(CNC(C2(OC)CCC2)=O)C1 C(=O)(C(F)C(F)(F)F)NCc1ccc(CN(C(c2ncn(C(C)C)c2)=O)C)cc1 Nc1cc(F)c(C(N2CC3CCN(C(C4CCCCS4(=O)=O)=O)C3C2)=O)c(F)c1 c1(C(=O)NCC2CC(C)N(C(C3CCC(=O)O3)=O)C2)sccc1S(C)(=O)=O C(=O)(C1CCc2nccn21)NCC(C1CC1)NC(C1CCOC1)=O.c1(N)ccccc1 Cc1ccc(C(N2CCC3C(NC(=O)CCOC4CCC4)CC23)=O)cc1CO Cc1n[nH]c2cnc(C(N3CCCC34CCN(C(C3COC(C)C3)=O)C4)=O)cc12 C1(C2CN(C(=O)CS(N)(=O)=O)C2)(NC(CN(C)C(=O)C2CC2)=O)CC1 c1(CC(c2nccs2)N(C(=O)C(=O)NC2CCOCC2)C)c[nH]c2ccccc12 N1(C(C(CC(=C)C)CC)=O)CCc2cccc(C(=O)OCC)c2C(C)C1 C1(C(=O)NCC(CC)(C)CO)CCCCCN1C(=O)CCN1CCOCC1 C(=O)(CCCCC(N)=O)NC1CC(CCNC(CC2(C=C)CCC2)=O)C1 c1(NC(=O)NC(C)CCN2CCOC2=O)cc(-c2ccccn2)n[nH]1 Cc1nc2cccc(C(=O)NC(C3CCCC3)CNC(=O)C(C)S(N)(=O)=O)c2[nH]1 c1(OCC)ccc(-c2nc(C3CN(C)CCO3)nn2C2CCCCC2C)cn1 N1(C(C(CCSC)NC(C2OCCC2(C)C)=O)=O)CC2CC=CCC12 C1(CC(=O)NCCC2CCOC2)CN(Cc2nccs2)CCO1 C1(NC(c2c(C)ccn2C)=O)(CNC(=O)CC2CCCC(O)C2)CCCCCC1 C1(NC(C2N(N=O)CCC2)=O)CC2CC1N(C(=O)CCOc1ccc(Cl)cc1)C2 N1(C(CC(C=C)CCC)=O)CC(C)CN(C(=O)CNC(N)=O)C(C)C1 c1(C(=O)NCC2(F)CCC(CNC(C(C)OC)=O)CC2)ccc2oncc2c1 N1(C(CC(C=C)(C)O)=O)CC2(C=C(C(=O)NC(C)C(C)SC)CO2)C1 N1(C(C2CC(=C)C2)C(=O)NCCCOC)CCS(=O)(=O)CC1 c1(C(=O)NCCN(CCOC)C(c2csnn2)=O)ccc(C)nc1 c1(C(=O)O)cc2ccccc2cc1C(=O)NCc1cc(Br)c(C2CC2)o1 C1(F)(C(=O)NCC2(C(=O)NC(C3CCCCC3)C(C)C)CCCC2)CC=CCC1 C1(NC(c2c(C)nc[nH]2)=O)CN(C(c2ncccc2Br)=O)CCC1F N1(C(C(CC)Nc2ccc(OC)cc2)=O)CCN2CC(c3cnccn3)CC12 c1(C(N2CC(CCNC(C(C)=C(CC)C)=O)OCC2)=O)cccc(C#N)c1Br CC1=CCN(C(C2CC(C)N2C(=O)C=Cc2cscn2)=O)CC1 N1(CC)CC(C(=O)Nc2cc(-c3ccc(C(=O)OC)cc3)[nH]n2)CC1=O C12(NC(c3ncoc3C3CC3)=O)CCCC1N(C(=O)CNc1cccnc1)CC2 N1(C(C2C(C(C)(C)C)CC2)=O)CC2(COC(CNC(c3cc(CF)on3)=O)C2)C1 N1(C(CN(C(C(C)OCC#C)=O)CC(C)C)=O)CC2(CCCO2)C1 c1(C(=O)NCC(CO)NC(CCNS(CC)(=O)=O)=O)ncoc1C1CCCCC1 Cc1nn(CCNC(=O)Cn2cc(-c3cccc(F)c3C)nn2)c(C)c1C C#CCCCCC(=O)N1CCN(C(=O)C(C)CC2CCCC2)C(C(C)C)C1 C1(NC(C(CCC)=CCC)=O)CCCN(C(c2cc(C)nn2C2CC2)=O)CC1F c1(C(N2CC3C(CNCc4ncc(C)s4)(C3)C2)=O)cccn2nccc12 c1(C(N(C2CCN(C(C3(CCOCC)CCC3)=O)C2)C)=O)cnc(OC)c(C)c1 c1(C(=O)OCC)cccnc1NC1CC(C)N(C(=O)COCC2CCOC2)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)C2CC=C(C(=O)N(CC(C)O)CCF)C1CC2 C(=O)(CCC(=O)c1cccc(N)c1)NC(C)(C)CNC(C1CC1C(F)F)=O C1(C(=O)NCC2(O)CN(C(c3ncncc3OC)=O)C2)(COC)CCC(=O)N1 c1(CC)nc(C)[nH]c1C(N1CCCC(CCNC(C2CCC2OC)=O)C1)=O c1(C(=O)NCC(CC=C)NC(c2csc(-c3ncc[nH]3)n2)=O)cnc(N)cn1 C(C(C)(CC1CC1)N=c1ccnc(CO)[nH]1)NC(C(n1cc(Cl)cn1)C)=O C12(CCN(C(=O)CC3CCC=CCC3)C1)C(=O)NC2.C(CO)(CCC1CC1)OC C12(C(=O)OC(C)(C)C)CCC(CC1)OC2.n1(CC(=O)O)nnnc1C c1(C(=O)NCC2C(NC(CC=C(C)C)=O)CCCC2)ccc2nccn2c1 N1(C(CCC(=O)N(C(C)C)C)=O)C2CCC1CN(C(C13CC(C)C1C3)=O)CC2 CCC(CC)(CC)N(C)C(CCC(C)NC(=O)CC1CC(C)(C)CO1)=O c1(C(N2CCC(NC(C(C)n3cccc3)=O)C2)=O)cccc(Cl)c1F C(=O)(C(CC(=C)C)NC(C1(CC)CC(C)(C)C1)=O)NCC(C=C)(C)C C1(C)(CC)C=C(C(=O)N(C(C)CN(C)C(c2sc(C)c(Br)c2C)=O)C)C1 c1(C(c2nnnn2CC(F)F)C(C2CCC2)C)cnn(C(F)F)c1.N N#Cc1cc(F)c(NC(c2cccc(-c3cccnc3)c2)=O)c(F)c1 C1(CCC)(NC(=O)C=Cc2ccc(C)s2)CCCN(C(c2ccc(Cl)cn2)=O)C1 C(CCCC(=O)NC1CCC(C(=O)NCCc2nccc(O)n2)C1)NC(N)=O Cc1noc(C)c1CNC(=O)COC(C)(C)CCNC(=O)CCc1ccoc1 C(=O)(C#CC1CCCC1)NCC1(CN(C(=O)CC(=O)N(C)C)C(C)C2CC2)CC1 c1(C(=O)Nc2cccc(C(F)(F)F)c2)cc(O)nc(Cl)c1.C12CC(C1)CNC2=O C(=O)(C1=CCCOCC1)NCc1c(NC(=O)OC(C)(C)C)nccc1 C1(CNC(C2C(=C)CC2)=O)CC2COCC2N1C(c1noc2c1COCC2)=O c1(OC)ccc(CNC(c2ncoc2CNC(=O)COC(C)=O)=O)cn1 c1(CC(N2CC(C)CC(NC(C(CC)SC)=O)C2)=O)cccc2sccc12 n1(C(C)C)ncc(C(N2CCC(C)(NC(C3CC(F)C3)=O)C2)=O)c1C1CC1 Nc1cc(F)cnc1C(=O)NCCC1(O)CCN(C(C2CCCCNC2=O)=O)C1 C1(C(C)NC(C(=O)NCC)=O)CCN(C(c2csc(CC(F)(F)F)n2)=O)C1 C1(CNC(=O)Nc2c(C)cccc2)CCN(C(C2CCC3CC3C2)=O)C1(C)C N1(C(C(C=CC)O)=O)CCN(C)CC1CNC(c1c[nH]c(Br)c1)=O C(C(CC(F)(F)F)NC(C1(O)CCSC1)=O)NC(COC(CC)C)=O c1(C(N2CC(OCC(=O)NCC3C4CCCC34)C2)=O)cnc(S)nc1 C1(C(=O)NC(c2nc[nH]n2)CC)CC(C)CCN1C(=O)CCC(=O)OC C1(NC(C(C)NC(=O)NC)=O)CCN(C(c2ccn(C)c2C(C)(C)C)=O)C(C)C1 O=C1NCCN2CCN(CC3CCCCC3(F)F)CC12 CC1CC(C)(C(=O)NC2CN(CC(=O)NC3(n4cnnn4)CC3)C2)C1 C1(CNC(C2C(CNC(C(CC)n3ccnc3)=O)CCO2)=O)CCC(C)=C(C)C1 c1(OCC)ccsc1CNC(c1coc(C)n1)c1nnnn1CCCSC C1(NC(CCCOCC)=O)CN(C(=O)Cc2c(O)ncnc2O)C2(CCCC2)C1 Cc1cc(C)c(NC(=O)C(=O)NC2CC3CCC2N(C(=O)CC(C)C)C3)cc1C C12CCC(C1)NC2.C1(CCC2CN(C(=O)OC(C)(C)C)C2)CCC(F)C1 c1(C(N2CC(C)C(C(N3CCC(O)(CF)CC3)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCC2N(C(c3cc(C)[nH]c3)=O)CCC2C)n[nH]c2c1CCCCC2 Cn1nccc1COCC(N1CCCC1CNC(=O)Cn1nnc(=O)[nH]1)=O c1(-c2n(C(CC)C(O)C(=O)N3CCN(C)C(C)C3)ccn2)ccc2c(c1)CCC2 N1(C(c2cc(OC)ncc2)=O)CC2CCN(C(=O)C(C)(C)O)C2C1 c1(C(=O)NC2CCC(CNC(COCCCCC)=O)CC2)ccc(C)c(C)c1Cl C(=O)(C(O)C1CCCC1)NC(CNC(=O)COC1CCC1)CO C1(N(C(=O)Cc2cnoc2)CC#C)CCN(C(=O)C=Cc2cnc[nH]2)CC1 N1(C(C(C=C=C)C)=O)CCC2(CCN(C(=O)CCCCOCC)C2)C1 C(=O)(C(C)(C)CO)NCC(CN(C(C1(CC)CCOC1)=O)C)O c1(CC)nn(C)c(Cl)c1C(=O)NC1C2CCN(C(=O)CCC3CCOCC3)CC12 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C)CC1CN(C(C2CC2Br)=O)C1 c1(C(N(C)CC2CCCN2C(C2CC2(C)C)=O)=O)cc2c(N)cccc2[nH]1 c12cccc(c1)C(=O)N2.C1(C(=O)NCCN(C(=O)OC)C2CC2)C(C)C1C N#CC1(C(N2CCCOC(CCNC(C3CCS3(=O)=O)=O)C2)=O)CCSCC1 c1(C(=O)NCC2CCC(NC(C(C)(C)OCC)=O)C2)cn2ccnc2s1 CN1Cc2ccccc2C(NCC(c2ccccn2)(C)C)C1=O c1(NC2CCN(NC(c3ccc(C)cc3)CCO)CC2)ccc([N+](=O)[O-])cn1 c1(C(=O)NC2(CF)CCN(C(CCC)=O)C2)ccc(P(C)(C)=O)s1 c1(NC(CC(C)(C)OC)C)cc(S(=O)(=O)NC(c2nnc(C)s2)C)ccc1C#N C1(c2cn(CCC3CC(N)C3)nn2)(C(C2CC(C)(F)C2)=O)CCOC1.CO C1(CNC(C2CC(C)C2)=O)CN(C(=O)C2=CCSC2)CCCO1 c1(OC)ccc(CC(=O)NCCCCCNC(c2cnnn2C)=O)nc1 C1(COC)(CNC(=O)C(=Cc2cscn2)F)CCN(C(c2ccoc2Cl)=O)C1 c1(NC(C)=O)cccnc1C(=O)NC(C)CN(C(=O)CC1CC(F)C1)C Cc1cc(NC(C2CC3CC3N2Cc2cccc(CO)c2)=O)cnc1C N1(C(C2C(C(C)O)C2)=O)CCCC(NC(=O)Cc2cccs2)C1C C1(C(N2CC(NC(C3(CC)CC3)=O)C(OC)C2)=O)CN2CCN1C(C)C2 c1(C(=O)NCC23CC(NC(c4cn(C)nc4C(F)F)=O)(C2)C3)ccc(F)c(F)c1F Cc1cc(I)ccc1CNC(=O)C(N1CCCC1c1sccc1Cl)=O CC(C)CCCC(C)CN(C(=O)CC1CCN1C(=O)CC(C)(C)C#N)CCO c1(OC)ccc(C(=O)NC2CC(CO)N(C(c3snc(C)c3N)=O)C2)cc1C c1(OC)ccc2[nH]c(C(=O)O)nc2c1NC(c1snc2ccc(Br)cc12)=O c1(C(=O)NC(CCCNC(c2n[nH]c(C)c2Cl)=O)C)c[nH]c2c(Cl)cccc12 C(=O)(C1=NN(CC)C(=O)CC1)NCC1C(NC(C(C=C)(C)CC)=O)C1 N(C(=NCc1cccc(N(C)C)c1)NC1CN(C)CC1O)C(c1ccccc1)C N1(C(=O)Nc2ccc(C)cc2)CCCC2(C1)CN(C(c1cc(C)no1)=O)C2 C(=O)(C(C)(COC)CC)NC1(CC=C)CCN(C(=O)C(F)n2cccn2)C1 Cn1cc([N+](=O)[O-])c(C(=O)NCC2(C)CCN(C(C3(C)CCC(=O)C3)=O)C2)n1 N1(C(c2ccc(OC)s2)=O)CCC(C)(C)C1CC(=O)NCC12CCCC1CCO2 C1(CNC(=O)CSc2n[nH]c(O)n2)C2CCC(C2)N1C(=O)Cn1cncn1 N1(C(c2c(C)nn(-c3ccccc3)n2)=O)CCCC(NC(=O)C(C)(C)F)C1C N1(C(CNC(CCNC(C)=O)=O)=O)CCCC(O)(CNC(C2(C)CC2(C)C)=O)C1 O=C(CC=C(Cl)Cl)N1CC2CC1(C(=O)NC1CSC1)C2 C1(C(=O)Nc2n(CC)ncc2)CC(F)(F)CN1C(c1cc(O)ccc1Br)=O c1(CN2CC(C(=O)Nc3nc(O)cc(OC)n3)OCC2)c(Cl)ccc(F)c1F N1(C(C2CC(=C)C2)=O)CCCCC1C(=O)NCC(C1CCC1)OC C1(F)(C(=O)NCC2(O)CC(C)(C)C2)CCCN(C(=O)CC(O)C2CCCC2)C1 C(C(C)(CNC(=O)CCCC1(NC(c2c[nH][nH]c2=N)=O)CCC1)CO)OC c1(-c2cc(C)ns2)nc(-c2cccc(Cl)n2)nn1CC(C)(C)C c1(CNc2nccc(C(=O)N(CCc3cnc[nH]3)CCO)n2)ccc2cncn2c1 C(=O)(CCC(C)(C)F)N1CC(N(C)C(c2csc(C3CC3)n2)=O)C(F)C1 Cc1ccc(C(N2CC3(CNC(=O)CC4CC4C)CCC2CC3)=O)c(Cl)c1Cl Cc1cc(CNC(=O)C(=O)N(C)Cc2sccc2Cl)n(C)n1 N1(C(CC(C=C)(C)C)=O)CCCC1C1CCCN1C(=O)C(=O)c1cccs1 Cc1ccc(-c2nc(C(=O)NC(C)C(N3CCOCC3)C)cs2)c(C)c1 c1(C(N2CCC(C)C2)=O)nnc(-c2cn(C)nc2-c2ccccc2)n1C1CC1 c1(CCC(=O)NCC2(COC)CN(C(c3csc(C)n3)=O)C2)nnc(O)nc1O C1(C(OC)(O)OC(C)(C)C)CC2(C1)CC(C)C2.C1(CO)CCCOC1C.C1(C)CC(O)C1 N1(C(C(c2cncc(F)c2)C)=O)CCCC(C)(NC(c2cnc(O)cc2O)=O)C1 N1(CC)CC(NC(=O)N(C)CC2CC3CN(C(=O)OC(C)(C)C)CC23)CCC1=O Cc1cc(C)c2c(c1)C(N(C(=O)Nc1ccc(F)cn1)CCO)CCCO2 N1(C(CC(C=C)CC)=O)CCC2CCN(C(c3cncn(C)c3=O)=O)C2C1 c1(OCC)cc(C(N2CCC(C(=O)NCC3(CO)CCC3)C2)=O)ccc1OC C12(C(N3CC=CC(C(N4CCC(CO)C(O)C4)=O)C3)=O)CCCC1CCC2 C(=O)(CCCS(N)(=O)=O)NC(CC)CN(C(=O)CC1COC(C)(C)CO1)C C1(C(N2CCC(C3OCC3(F)F)CC2)C(=O)NCC(=C)C)CC2CCC1CC2 C(=O)(C1=CCC(F)(F)CC1)N(C(C)C(c1ccc2c(c1)OCO2)=O)C c1(C(=O)NCC2C(NC(C(C)OCC)=O)CC2)cnc(Br)s1 N1(C(c2scc(C)c2Cl)=O)CC(NC(C2CC3C(C2)C3(F)F)=O)CC(C)C1 c1(SC)ncc(N)c(C(=O)NC2CN(C(=O)CC3C(=O)NN=C3C)C2)n1 O=C(C1CSc2ccccc21)NCC1(F)CC(NC(c2ncccc2O)=O)C1 N1(c2ccc(C(=O)NC3C(=O)NCCCC3)cc2)Cc2ccccc2C1=O C(=O)(CC(C)CC(C)(C)C)NCc1nccc(C(=O)NCC(C)OC)c1 c1(CC)ccc(F)cc1NC(=O)CC(C)(C)NC(=O)CN(C1CCC1)C C1(NC(=O)Cc2ccn(C(F)F)n2)CC2CCC1N2C(=O)C(O)Cc1cnc[nH]1 C1(O)(CCNC(CC2CC(CC(=O)O)C2)=O)CCNC1 c1(OCC(=O)NCC2CCN2C(=O)CC2CCCCO2)ccc(C(F)(F)F)cc1 C#CC1Cc2ccccc2C1NC(=O)NNC(=O)CSc1nc2ccccc2[nH]1 c1(OC(CN(C)C(=O)NCC2(CC3CC3)CC2)=O)ccccc1 N1(C(c2cc[nH]n2)=O)CCN(C(c2cc(O)ccc2Cl)=O)C2CS(=O)(=O)CC12 CC1CCC(NC(c2cccnc2CO)=O)CN1C(C1C2CCCCN12)=O C(=O)(CC(C)(C)O)NC(C(=O)NC(c1c(C)ncs1)C)c1ccoc1 C1(NC(=O)CCc2cn[nH]c2)CC2CCC1C(NC(=O)CSC1CC1)C2 N#CC1CN(C(c2ccc(C(F)(F)F)cn2)=O)CCN1C(=O)CN1CC2CC2C1 CC1=NOC(CC(=O)NCc2ccsc2C(=O)NOCC2CCCO2)C1 C1(N(C(CC(C)SC)=O)CC2CC2)CCN(C(=O)C(C)NC(=O)C(C)(C)C)CC1 C12CN(C1(C)C)C(=O)C(C)(CO)OC2.C12(C(=O)OC)CCCC1C2 N1(C(CNC(CCC)=O)=O)CCCC(C)C1CCNC(c1nc(C2CC2)cs1)=O C=C(C)CN=c1[nH]c(=NCCc2nc(C(C)(C)C)cs2)c2sccc2[nH]1 C=C(C)C1OCCC1C(N1CCCC(NC(c2cnc(C(C)(C)C)o2)=O)C1C)=O c1(OC)cc(NC(C2CCCN2C(c2ccc(CO)o2)=O)C)ncn1 N1(C(CC(CNC(C2C3CN(C)CC32)=O)(C)C)=O)CC2CCC(C1)C(=O)O2 c1(C(=O)NC2CCN(C)CC2)ccc2nccn2c1 C12(CNC(c3[nH]cc(C)c3C)=O)CN(C(c3cn(C4CC4)cn3)=O)CC1CCO2 CC1(C)CCOC(CC(=O)NCC#CCNC(c2ccncc2Br)=O)C1 c1(C(=O)NC2C(CNC(c3cc(C(N)=O)oc3)=O)C2)cc(C2CC2)[nH]c1C1CC1 C(=O)(CCCCNC(C1OCCC1C)=O)NC(COCC)(C)C C(CC(C(=O)N1CCOC(CCF)C1)NC(=O)CC1(CS(C)(=O)=O)CC1)SC CC(C)CC(CNC(=O)C(C)n1cccc1)C(=O)Nc1cc(F)ccc1O C1(C(CC(=O)NCCN(C(=O)C(C)(C)c2ccnn2C)CC)C)CCCC(=O)N1 C(=O)(C(C(C)C)C(C)C)NC1C(C(=O)NCC(CSC)(C)C)CCCC1 CC(C)CCCCCC(=O)N1C2CCC1CC(CNC(c1cnn(C)c1F)=O)C2 c1(C(CCC)=O)ccccc1OC(=O)NNC(=O)C1COCCO1 c1(OC)ccnc(N(CCNC(c2sc(C)nc2C)=O)CC)n1 C(CC(=O)NCCCOC1CCC1)(C(F)(F)F)NC(COC(C)=O)=O Cc1nc(C)c(C(N2CC(NC(=O)Cc3ccc(C(C)C)cc3)C(F)C2)=O)s1 n1(CC(N2CC(OC)C(NC(C3CC(SC)C3)=O)C2)=O)nc(C)c(C)c1C c1(CN2C(C(=O)Nc3nc(C)nc(Cl)c3)CC(C)C2)ccc(C)c(C#N)c1 N1(C(C2CCC(N(C)C)C2)=O)CC2=C(C1)CN(C(C1(C)CC13CCC3)=O)C2 N1(C(CC2N(CC)CCOC2)=O)CC=C(CCNC(C2CCSC(C)C2)=O)CC1 CCC(C)(CO)NC(=O)C(C)OCCNC(=O)COc1ccccc1.C1CO1 N1(C(C2CCN(C(C)C)CC2)=O)CC2(CCN(C(C3COCCOC3)=O)C2)C1 C(=O)(C1CCOc2ccccc21)NC1C2OCC(NC(=O)COC3CCC3)(C2)C1 CC(C)(F)C(=O)NCc1cc[nH]c1C(=O)NC1(c2cccs2)CC1 c1(C(N2C(CN(C(=O)C3=CCCCO3)C)CCCC2)=O)nccc2cc[nH]c12 N1(C(C(C=C)c2ccccc2)=O)CCC(CO)(Nc2ncnc(C(C)C)n2)CC1 C(=O)(C(C)CC(C)(F)F)NCCCCC(C)NC(=O)C(C)(C)CF c1(CC(C(=O)OC)NCC(O)COCC(F)(F)C(F)F)cc(Cl)ccc1O N1(C(C=CC=CCC)=O)CCC(C2CC2)(NC(C23CCCC2C3)=O)C1 N1(C(C2N(C(=O)OC(C)C)CCC2)=O)CC2CC1C2NC(=O)Cc1cn(C)cn1 N1(C(C(C)=CC)=O)CCn2ncc(CNCCC(=O)N(C)C(C)=O)c2C1 c1(CCCCCC)nc(-c2cc(=O)cc[nH]2)n(-c2ccc(C(CC)OC)cc2)n1 N1(C(C=CC=CC)=O)CCCC(C)(NC(=O)CSc2nccn2C)C1 c1(C(N(CC(C)NC(C2(C(F)(F)F)COC2)=O)C)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C#CC1CCN(C(=O)CC2CCC(NC(=O)CN(C)C(=O)OC)C2)C1 N1(C(C(=C)C(F)(F)F)=O)CC2(CCOCC2C(N2CC=CCC2C(N)=O)=O)C1 c1(C(C(=O)Nc2ccc(F)cc2)N(C(C#C)C2CCC2)C)cnc(C)c(C)c1 CCC(F)(F)C(C)(C)CNCc1ccc(C#N)cc1F c1(C(=O)NC(C)CNC(C2(C)CCCCNC2=O)=O)cc(F)c2c(c1)CCC2 C1(C(=O)Nc2cccnc2O)CC2(CCN(C(c3cccc(=O)o3)=O)C2)C1 C1(NC(c2cncc(C)c2)=O)COC2(CCN(C(=O)CC3(O)CCCC3)C2)C1 c1(C(=O)NCC(CNC(C(C)CC2CC2)=O)(C)O)cn(C)nc1-c1ccnn1C CC1CCCN(C(C2CC2NCc2nc(-c3ccccc3)no2)=O)C1 c1(OC)cncc(Br)c1C(=O)NCCN(C(=O)CCCOC(C)C)C c1(OC)c(C)nc(SC(=O)N=c2ccc(-c3ccc(Cl)s3)n[nH]2)nc1C CON1CCC(CC(=O)NCC2(CNC(=O)C(F)CC3CCOCC3)CC2)CC1 CCC(CC(=O)NCC1CCN1C(=O)COC1CCC(C)CC1)SC Fc1cncc(C(c2nnnn2-c2ccccc2)NCC2CCCSCC2)c1 c1(CC)cccc(CN=C(NCC(=O)N(C)C)NCC2CCC2)c1 CS(=O)(=O)C1CC(C(N2CCC3C(NC(c4ccc(Cl)o4)=O)CC23)=O)C1 CCC(CC(=O)N1CC(C(=O)NC(C2CC(F)(F)C2)C)C(C)C1)C(C)C C1(CNC(C2(CC)CCCO2)=O)CN(C(c2csc(C(F)(F)F)c2)=O)CC1C S(=O)(=O)(c1ccc(C(C)(C)C)cc1)NC(C1CCCCO1)COCCC(C)C c1(C(=O)NC2(C(C)C)CCCCC2)cc(=NCC(C)(C)c2ccn(C)n2)[nH]cn1 CC(CC(F)F)C(=O)NCCC1CCN(C(c2cc(C3CC3)no2)=O)C1 C1(NC(C2CC(=O)NCC2)=O)CC2CC1N(C(C1COC1)=O)C2 c1(C(=O)NCC(CC=C)NC(c2ccn(CCO)c2C)=O)cccc2nncn12 Cc1[nH]nc2cc(C(=O)Nc3cccc(C(C)(C)C)n3)ccc12 C1(NC(=O)C2=CSCCO2)CC2(CCN(C(c3cscn3)=O)C2)C1 C1(C(N2C(C)CN(C(C3CC(C4CC4)C3)=O)CC2)=O)CN=C2N=CNN2C1 Cc1ncc(N)cc1C(=O)NCC1CCN1C(c1ccc(C(F)F)nc1)=O c1(C(C(=O)N2CC(N(C)C)C2)NC(C(N2CCNC2=O)C)=O)ccccc1 Cc1ccncc1CC(N1CC(CN(C)C)C1)=O.c12ccc([nH]1)C(=O)NC2 c1(C(=O)NC(CNC(=O)CCc2cncs2)CO)cccc(C(F)F)c1Cl n1(CC(=O)NC2CC[Si](C)(C)C2)c(C(=O)O)cc2ccccc12 C1(NC(c2ccc3oc(O)nc3n2)=O)CCCC12CCN(C(=O)Cn1cccn1)C2 CN=c1ccc(Br)c(C(N2COCCC2C)=O)[nH]1 C1(C(=O)NC2(CO)CN(C(c3c(CC)nccc3)=O)C2)CC2CCCCN2C1 C#Cc1c[nH]nc1C(=O)NCC1C(NC(=O)CCSCc2ccc(Cl)cc2)C1 C(=O)(C(C)(C)CS(N)(=O)=O)NCC1C(NC(c2c(C)nc(-c3cccs3)cc2)=O)C1 CCC(N=c1[nH]c(=NCCC(C)OC)c2ncccc2[nH]1)C(C)C Cc1ccc2nc(C(=O)NC3(C)CCN(C(C4CCCC45CC5)=O)C3)cn2c1 c1(NC(c2ccc(NC(c3scc(COC)n3)=O)cn2)=O)ccc(Cl)c(CO)c1F C(=O)(C(F)(F)C(F)F)NCCCCCCN(C(C(N1C(=O)CCC1=O)C)=O)C CC(C)(CNC(C1CC(CC2CC2)C1)=O)CC1CN(C(c2sccc2F)=O)C1 CC1CCN(CC(c2ccc(F)cc2)NC(=O)N(C(=O)C(O)c2ccsc2)CC)CC1 CC1CN(C(=O)C=CC(C)NC(C2(O)CCOCC2)=O)CC(=O)N1 c1(C(CC=C(C)C)C)nc(-c2ccnn2C)nn1C1COC(C)(C)C1 N1(C(Cn2cccc(C)c2=O)=O)CCC2CC1CN2C(c1cc(C#N)cc(C)n1)=O N1(C(c2ccc(CC)[nH]2)=O)CCC(C)C1CNC(=O)C=C1CCCC1 C(=O)(CS(=O)(=O)c1ccccc1C)NC(CNC(C(S(CCC)(=O)=O)C)=O)C C#CCC(CC#C)C(=O)NCCOCCNC(=O)C(C)(C)C1CC1 C(=O)(C1=C(C)CCC1)OC.N1(C(=O)OC)CCCCC1CCC1c2nc(n[nH]2)N1 O=C(C1CCCc2nc[nH]c21)NC1CCN(C(c2ccnn2CC(F)(F)F)=O)C1 CCC(C)C(C(=O)NCCn1cc(-c2csc(C3CC3)n2)nn1)c1ccccc1 c1(C(=O)NC23C(CN(C(C4=C(C)CC4)=O)C2)CCC3)ccc(S(N)(=O)=O)c(C)c1 c1(SC)ccc(N)cc1C(=O)NCC(C1CCCCC1)NC(=O)C(O)CN(C)C C=CCC(C)(C)C(=O)N(CCC(=O)N1CC(F)CC1C)OC CC1CN(C(c2ccco2)=O)CC1NC(=O)CCc1ccc(O)nc1 C1(COC)(NC(C2CC3CCC(C2)O3)=O)CCCN(C(C2(C(C)C)CC2)=O)C1 CC1(C)CCCN(C(C2COCCN(C(=O)CC34CCCC3C4)C2)=O)CC1 Cc1nc(C2CC2)oc1C(=O)NC1CCCC(CNC(=O)CC(C)N(C)C)C1 c1(SC)cc(C(=O)NCC(C)(O)CNC(=O)CC(O)CN(C)C)ccc1N c1(C(c2n(CCSC)nnn2)NC(c2ccccc2F)C)cnc(C)c(C)c1 N1(C(C(C)C(F)F)=O)CC2CCC1C1CN(C(=O)C=CS(C)=O)CC21 C(=O)(C(Cn1cccn1)NC(C1(CC)CN(C(C2OCCC2C)=O)C1)=O)OCC O=C(C#CC1CCC1)N1CC(OCCNC(C2CCCN2CCCO)=O)C1 N1(CC(=O)NC(C2CCCCC2)C)CC(=O)CC(C)C1 c1(OC)ccc(C(=O)NC2CC(NC(C3(CN(C)C)CCC3)=O)C2)c(F)c1F C(=O)(CC(C(F)F)n1ccnc1)NC1(CNC(C=CCCC)=O)CCOC1 c1(N(C(C2CCCNC2)C)C(c2ccnc(Cl)c2)=O)ncnc2[nH]cc(I)c12 c1(NC(C2(C(=O)Nc3cccc(OCC)c3)CC2)=O)ccccc1S(=O)(=O)F Cc1cn2c(C(=O)CSC3CN(C(C)(C)C)CCCO3)csc2n1 Cc1ccc(C(C)O)cc1NC(=O)NC1CCN(CCF)C1=O C(=O)(C(C)N=c1cc[nH]cc1)N1CC(C(=O)NC(F)(F)C(F)(F)F)(CC)C1 c1(C(N2CC(C(C(N3C(CCC)CCC3)=O)OC)C2)=O)ccc2n[nH]cc2c1 C1(NC(c2cn(CC)nn2)=O)CCC(C(N2CCC2CF)=O)CC1 c1(C(N(C(CCNC(C=Cc2c(C)ccs2)=O)C)C)=O)coc2c(F)cccc12 C1(NC(c2c(C)nco2)=O)CCN(C(=O)C(c2ccccc2Cl)O)CC1F C=C(C)CC(C(=O)NCc1nnnn1C)NC(c1cscn1)=O C1(N(C(=O)OC(C)(C)C)CC)CCN(C(=O)OC)C1C(F)(F)F C(=O)(CCCC(=O)N1CCCC1(C)CNC(C1CC12CCOCC2)=O)N(C)C c1(NC(C2C(NC(CCC(C)C)=O)C2)=O)cc(Cl)c(C#N)cc1Cl C=Cc1ccc(C(N2CC(CC(=O)NC3(C)CCC(C)CC3)C2)=O)cc1 C(c1cscn1)=CC(=O)NCCN(CC(C)O)C(=O)CC1CCCN1C CCN=c1ccc(C(N2CCC(NC(C3CC(=O)N3)=O)C(F)C2)=O)c[nH]1 c1(CC(=O)NC2C(NC(C=CCC)=O)CC2)nocc1C c1(C(=O)NC2C(OC)CN(C(CCCCC=C)=O)C2)ccc2c(c1O)CCCC2 CC(CCC(C)(C)C)C(=O)N1CCC2(C(=O)NCC3(CN=[N+]=[N-])CC3)CCCC12 C(=O)(CC(C)CC(F)(F)F)N1CCC(C)C(NC(c2cc(C)cc(C)c2)=O)C1C CC1CCCC(C(N2CC3CC2C2CC32)C(=O)NCc2ccccc2Br)CC1 C(=O)(CC1CCc2ccccc21)NCC1(CNC(CC(C)OC)=O)CC(F)(F)C1 N1(C(C=COCC)=O)CC(NC(=O)C(N2C(=O)CCC2=O)C)CC(C)C1 C#CC1(NC(C2(F)CCN(C(=O)CN(C(=O)C(C)C)C)C2)=O)CCCOC1 n1(CC)c(C)cc(C(=O)NCC(C2CCC2)NC(c2ccc(C)cn2)=O)c1C N1(c2ccnc(N(CCCC(=O)NC)C)n2)CCS(=O)(=O)CC(C)C1 c1(C(=O)NCC2C(CNC(c3c(C)cnn3C(C)C)=O)C2)cccc2ccsc12 Cc1ncnc(N2CCC(C)C2CNC(c2cscc2C)=O)c1C#N CCC(C(=O)NCc1cc(C(=O)NC2CC(C)(C)OC2(C)C)ccn1)C(F)(F)F c1(C(=O)NC2(CC)CCN(C(C(C=C)(C)C)=O)CC2)cc2c(nc1O)CCSC2 c1cccc(F)c1Cl.C1(N(CC(F)F)C(C2C(C)C2)=O)CC2CNC1C2 Cc1c(C(=O)NC2CCN(C(=O)C=CCn3cncn3)CC2O)ccc(F)c1F CCCCS(=O)(=O)CC(=O)NC1CCN(C(=O)C(c2ccccc2)C)CC1CO C(=O)(C1CCCc2cncn21)NCCOCCN(C)C(C1(C)CC=CC1)=O c1(OC)cnc(C(N2CC(OCCNC(C3CSCCS3)=O)C2)=O)cn1 C(=O)(C(C)(C)CCF)N1C(C)CC(CNC(C2(COC)COC2)=O)C1 C=C(C)CC(C)C(=O)N(C1CCN(C(c2cc(SC)oc2C)=O)CC1)CCC C1(Nc2c(C)c(NC(Cc3ncnn3C)C3CC3)ncn2)CC2(COC(C)C2)C1 CCC1=NOC(CC(=O)NCCC2COCCN2C(=O)CN(C)C(=O)C2CC2)C1 N1(C(C(C)NC(=O)C(N)=O)=O)CCCCC1Cn1cc(-c2cccnc2F)nn1 N1(CCCOC)CC(C(=O)NCc2ccc(OC3(C(F)(F)F)CC3)cc2)CC1=O.COC C1(F)(C(=O)NCc2nn(C)c(=O)o2)CCCN(C(=O)C(C2CCCCC2)F)C1 c1(C(=O)NC(C)(CNC(c2ccncc2C2CC2)=O)CO)ccc(F)cc1F c1(-n2cc(CCCCNC(C3(F)CC3)=O)nn2)ccc(O)cc1 N1(C(CCC)=O)CCC(CN(C(=O)COc2ccc(Br)cc2)C)CC1 N1(C(c2cc(C)oc2C)C(=O)NCCC)CCN(C(=O)C(F)(F)F)C2(CC2)C1 N1(C(C(C(C)(C)C)SC)=O)CC2(CC(NC(=O)C=Cc3cnccc3C)CO2)C1 C1(C(N2CC3C(C(=O)NCc4cc(C)sc4C)(C3)C2)=O)CC(C2CC2)=NO1 C1(C(N2CC3(CC(NC(C(F)=CCC)=O)C3)C2)=O)(OC)CCC(C)(C)CC1 N1(C(C2(NC(=O)C(F)C3CCCC3)CCSC2)=O)CCOC2CCC12 C1(C(N(C)CCN(C(=O)C(=Cc2cccc(F)c2)F)C)=O)CNC(=O)CC1(C)C C=CCCCC(=O)N1CC2C(CNC(c3ccccc3NS(=O)(=O)CC)=O)C2C1 C(=O)(C1=CCCOCC1)NC(CNC(C1N(C(C)(C)C)CC1)=O)C1CC1 CC1CC(NC(=O)CC23CCC(CC2)C3)CN1C(=O)CC(=O)NCC1CC1 Cc1ccc(-c2cn(C(C)C)nn2)c(C)c1.C1CCN(C(=O)CN(C)C)C1C(C)C C(=O)(CCCCCCCC(=O)N(C)CCOCCNC(=O)CC1=CCCC1)OC C=CCN(OC)C(=O)CCNC(c1ccc(CO)nc1)=O c1(NC(C(C)Cn2ccnc2)=O)cnc(F)c(Cl)c1 c1(C(=O)NC2(C)CN(c3nc(C)c(C#N)cc3)C2)ccc2c(c1)C(=O)NCC2 c1(CC(=O)N(C(C)C)CCNC(c2ccoc2Cl)=O)cccnc1Cl C(=O)(C(C)C(O)C(C)C)N1CC(CCNC(c2nc(OCC)oc2)=O)C(C)C1 N1(C(CN(C(CN2CCC(C)CC2)=O)C)=O)CCC(N=[N+]=[N-])CC1 C1(NC(c2cc(C)c(C)s2)=O)CC2CC1CN(C(=O)CCC1CCC1)C2 N1(C(c2csc(-c3ccccc3Br)n2)=O)CCN(C(C2CC2F)=O)C2CC12 C1(CNC(C=CC(=O)OCCCC)=O)CCC(NC(=O)CS(=O)(=O)N(C)C)CC1 N1(C(=O)NC2C(OC)CCCC2)C2CCC1CN2C CC(C(=O)NCCCCNC(C1(Cl)CC1)=O)C(C)S(C)(=O)=O CCS(=O)(=O)CC(=O)N1CCCCC(CNC(c2sc(C)cc2C)=O)C1 c1(C(NOC(C(=O)OC)C)=O)cncc(CNC(=O)Cn2cncn2)c1 Cc1cc(C(N2CC(CNC(=O)CCc3ccn(C)c3)C2)=O)ccc1Br c1(C(=O)NCC(C)(O)CNC(c2nocc2C2CC2)=O)ccccc1C(F)(F)F c1(CNc2snc3cccc(C(=O)O)c32)nc2ccc3ccccc3c2[nH]1 C1(CC(=O)NCCC2N(C(c3ccc(OC)nc3)=O)CCC2)CCCNC(=O)C1 c1(C(N2CC(c3ccccc3)(NC(C3CC4(CCC4)C3)=O)C2)=O)cccnc1S Cc1cc(C(=O)NCc2ccc(C(=O)NCC3CCC(F)C3)cc2)cc(C)c1F C1(OC)(CNC(C2C=CCN2C(=O)C=C2CCC(C)CC2)=O)CCCCC1 C1(C(N2C(C)(CC(=O)N(C(C(C)C)C)C)CC2)=O)CCC(C#N)CC1 c1(CCC)ccc(C(C(=O)NCC)N(C)Cc2ncoc2C2CCC2)o1 N1(C(C2(OC)CCC2)=O)C2CCC1C(CNC(c1cccc(C(F)(F)F)n1)=O)C2 c1(C(=O)NC(CC)C(=O)NCCN(C2CC2)CC)cnc(O)c(C)c1 N1(C(C(=O)NCCOCC)C)CC2CC(NC(c3cc4ccsc4s3)=O)CC1C2 c1(CNC(c2cncc(NC(C)=O)c2)=O)ccc(F)cc1OCCC(C)C C(=O)(CC(C)C=C)N(C1CCN(C(c2cc(C)nn2CC)=O)C1)CC#C c1(C(=O)NC2CCN(c3ncc(C)c(C)n3)CC2F)ccc(C#N)cc1F c1(C(=O)NCC(C)(C(C)C)NC(C2C(C=C)CC2)=O)cncc(OC)c1C c1(CC)cc(C)ccc1C(=O)NC(C1CCOC1)CNC(c1csc(F)c1)=O C=C(C)C(C)(C)C(=O)N(C1CCN(C(=O)C(c2cnn(C)c2)C)CC1)C c1(C(N2CC(F)(CNC(c3cn(CCC=C)nn3)=O)C2)=O)ccc(C)c(C#N)c1 c1(C(=O)NC2C(NC(c3csc(CC(F)(F)F)n3)=O)CCC2)ccncc1O N1(C(C2(C=C)CCC2)=O)CCCC(N(C)Cc2noc(COC)n2)C1 C1(CC)CN(C(=O)CC(C)(O)COC)CCN1C(=O)CCc1ccn(C)n1 CC(CC(=O)NC1CCCCC1NC(=O)CCNC(=O)C(C)(C)C)P(C)(C)=O CCC(C)(C)C(C)CC(=O)N1CC(NC(=O)C=Cc2ccn(C)c2)CC12CCC2 N1(C(CC2CCN(C(CCCOCC)=O)C2)=O)CCC(O)CC1C1CC1 C1(NC(c2c(C)cc[nH]2)=O)C2CCC(C2)C1C(=O)NC1(CCO)CCOC1 C1(C(N(CC(C)OC)CC)=O)(NC(c2ccc(C(F)F)o2)=O)CCSC1 c1(CNC(c2c(OC)n(-c3ccccc3)nc2)=O)cc(Cl)c2ccncc2n1 C1(C(=O)NCCC2C(C)OCC2)CC12CCOc1ccc(F)cc12 c1(C(=O)NCCCCC(C)NC(=O)Cc2cc[nH]c2)ccccc1N=[N+]=[N-] N#CC1(C(=O)NCC2(NC(c3occc3F)=O)CCCC2)CCCC1 Cc1ccc(F)c(C(N2C(C(=O)NC3COCC3CO)CC3CC23)=O)n1 N12CCN(CC1)CCCNC(=O)C1CC1CC2=O.C1(C)(CC)CS(=O)(=O)C1 c1(CC(=O)NC2CCC(C)(NC(C(CCC)OCC)=O)C2)ccc2nsnc2c1 N(C(=NCCCSC)N1CCC2(CCCCCC2)C1)CC(CC)CO C1(NC(c2c(OC)n[nH]c2)=O)CC2CC1CN(C(c1cc(O)ccc1Cl)=O)C2 C(=O)(C1CCc2ccccc21)NC1C(C)(C)CN(c2ncncc2I)C1 c1(C(=O)NC(CC=C)CNC(c2cnn(CCO)c2)=O)ccc2nnnn2c1 N1(C(C2(CC#C)CCCO2)=O)CCC(NC(=O)Cc2cccc(OC)c2)C(O)C1 C(C(C)CC(=O)NC1C2CC1N(C(=O)Cn1nnnc1-c1ccsc1)C2)OC O=C(CC1=CCOCC1)NCC1(F)CCCN(C(c2ccc(C(F)F)o2)=O)C1 Cc1ccc(C2(CNC(=O)CNC(=O)CCc3cnco3)CC2)nc1 C1(NC(C2CN(C(c3cnc(C)nc3)=O)C(C)(C)C2)=O)CCOC2(CCC2)C1 CN1CCC(C(N2CCCC(N(C(=O)CCN(C)CCO)CCO)C2)=O)CC1 c1(N2CCC(N(C)C(C3CCCCS3(=O)=O)=O)C2)nc2c(cc1Cl)C(=O)OC2 c1(C(=O)NC2CCC2CNC(C2CCS(=O)(=O)N2)=O)cc(Cl)ncc1O c1(OC)ccc(S(=O)(=O)N2CCN(Cc3cc[nH]n3)CC2)cc1-c1cccnc1 N1(Cc2ccn(CCC)n2)CCCC(C(=O)NC2CCNC2=O)CC1 C(CCCCC(=O)NC)=CCCC.N12CCN(C(=O)C(O)CCSC)C(C1)CC2 C12(Nc3ccc(C#C)nc3)CCC(c3nc(C4CC(O)CCO4)no3)(CC1)CC2 Cc1ccc(N)c(C)c1C(=O)NC1CCCC1CNC(=O)C(C)CC(C)C C1(NC(C(COC)O)=O)CCCCCC1NC(c1cc(Br)n(C)n1)=O N1(C(CCNC(=O)NC)=O)CCCC(N=c2cc(Cl)nc(COC)[nH]2)C1 c1(C(=O)NC2CCN(C(C(CCCC)CC)=O)C2C)ccc(C)cc1[N+](=O)[O-] c1(C(N(c2cn[nH]c2)CCC)=O)cc(-c2nn[nH]n2)c[nH]1 N1(C(Cn2c(C)ncc2)=O)CC(NC(c2cncc(C3CC3)c2)=O)CC1(C)C O=C(CC(O)C1CCCC1)NC1CCC1.C12CC(C1)C(F)C(=O)N2C1CCC1 c1(CN2CC(C(=O)Nc3cnc(C)c(Cl)c3)SCC2)c(C)ccc(C)c1O Cc1oc(-c2ccco2)nc1C(N1CCC(NC(C2OCCC2C)=O)C1)=O Cc1ccc2oc(=NCCC(C)NC(c3cnn(CCO)c3)=O)[nH]c2c1 N1(C(c2c(OC)nccn2)=O)CC(C(N2CC3(CC(O)C3)C2)=O)CC2OCCC12 N1(C(c2ccnc(COC3CCN(C)C3=O)c2)=O)CCC(O)CC(C)(C)C1 c1(CC)ccccc1C(N1CC(CC)CC1CNC(C1CC(C)(NC)C1)=O)=O C(=O)(C(CC)C(C)C)N1CC(CN(C(CCN(CCCCC)C)=O)C)OCC1 C1(CNC(CNC(COCC#C)=O)=O)CCCCC1CCC=C N1(C(c2c(N)csn2)=O)CCC(NC(=O)C(F)(F)F)C(F)(F)CC1 c1(NCCOc2cc(C)cc(C)c2)nccc(=NC2CCCC2C#N)[nH]1 c1(C(N2CC(=CCNC(CC3(C(=O)OCC)CCC3)=O)C2)=O)ccnn1COC C(CCC(=O)N1CCCC1C(=O)NC1(CN(C)C)CCC1)SC CC1(CNC(=O)C=Cc2ccc(F)nc2)CCN(C(C2CC=CC2)=O)CC1 C1(NC(C2C(OCC)C2)=O)COCCN(C(=O)C(C)(C)OC)C1 c1(NCC(c2ccccc2)OCCCC)nccc(=NCCc2sccc2Br)[nH]1 c1(CC(=O)OCC)csc(=NCC(C)NC(=O)C(F)(F)F)[nH]1 c1(C(=O)NCCC(C)(C)NC(CSCCC)=O)ccnc(S)c1 C1(CNC(CC(=O)OCC)=O)CN(C(=O)Cc2c(Cl)cnn2C)CC1C(F)(F)F N1(C(C2CC(C)(C)C2)=O)CCN(CCO)C(C)(C)C1 Cc1nc(C#N)c(NCCC(N2CCC(NC(=O)COC(F)(F)F)C(C)C2)=O)o1 CC1(C)CCN(C(c2cnccn2)=O)C(C(=O)NCC2COC(=O)C2)C1 N1(C(CC2N(C)CC=CC2)=O)CC2CC1CN2C(C1CC1CC(C)(C)C)=O C(CCC(C(=O)N(C)CC1(SC)CC1)NC(=O)CC1CCCCO1)OCC c1(C(N2CCC(NC(CC(=O)NCC#C)=O)C2C2CC2)=O)csc2ccccc12 CCC(C#N)C(=O)N1CCCC(C(C)(C)C(=O)NCC(N2CCCCC2)C)C1 N1(CC)CC(CNC(=O)CC2(C)CCN2C(c2ccc(C)n2C)=O)OC1=O CCC(C)C(=O)C(=O)NCC1(C(=O)NCCCSC)CCCO1 CCCCC(O)C(=O)NC1(C(=O)NCCC2CCCC23CC3)CC1 C1(C)(NC(C(CC(F)F)N(C(c2cnc(CC)nc2)=O)C)=O)CCCCC1(C)C c1(CCC)ccc(OC(C)C(=O)NC(Cc2ccnc(Cl)c2)C(=O)OC)cc1 O=C(C1CCCc2n[nH]cc21)N1CCC2(CC1)CN(C(C1CCCC(O)C1)=O)C2 Cc1cc(N2CCCC(OC(=O)N(C)C)C2)nc(N2CCOC(C)CC2)n1 C(=O)(C1=CCCOCC1)N(CCNC(c1ccc(F)cn1)=O)CC1CC1 C=C(Cl)CCC(=O)NCc1ocnc1Cn1cc(Cn2ccnc2C)nn1 C(=O)(CCCC(=O)NOC(C)(C)C)N(CCCCNC(c1c(C)sc(O)n1)=O)C c1(C(=O)NCC2(NC(C3C(F)(F)C34CC4)=O)CC2)ccc2nncn2c1 N1(C(c2c(C)c[nH]c2)=O)CCC(OC2CN(C(=O)Cn3cnnc3)C2)CC1 c12cc-1ccn2.c1(NC(=O)Nc2scc(C(=O)OCC)n2)[nH]c(C)nc1C N1(C(c2cnc(C)nc2)=O)CCC2(CC2C(=O)Nc2ccnc(C(F)(F)F)c2)C1 N#Cc1cc(Br)cnc1NCC1CCCCN1C(C1CC2(CCC2)C1)=O C(=O)C(C)Cn1ccnc1.C(CNC=O)SC N1(C(CC(C(=C)C)OCC)=O)CC2(CCN(C(=O)CN3CCC(O)CC3)C2)C1 N1(C(C(C2CCC2)OCC)=O)CCN(C(c2ccc(C#N)cn2)=O)CC1CO C12(CNC(C(C3CCN(C(CC=C(C)C)=O)C3)F)=O)CCC(CC1)C2 CC(C)(CCCNC(=O)C(F)C1CCC1)C(=O)NCC1(C)CC1F C1(C(=O)NC2CCC(CCC(=O)NCCC3CCCCC3)C2)CC(C2CC2)=NO1 Cc1cc(C(N2CCC(O)(CNC(C3CC(C(C)C)C3)=O)C2)=O)cc(C)c1 C1(CNC(CCCCOC)=O)CC12CCN(C(c1ccnnc1O)=O)CC2 c1(NC(CNC(CNCC(CC)OC)=O)=O)ccc(Br)cc1 N1(C(C(c2ccc(C)cc2)(C)C)=O)CCN(C)C(CNC(=O)C(CO)N(C)C)C1 Cc1nc2c(o1)CCN(Cc1ccc(S(C)(=O)=O)cc1F)C2 N1(c2cc(C)nc(C)n2)CCC2CC(C(=O)NC3CC4CC3C(O)C4O)C2C1 C(C(N=c1nc(OC)[nH]c(OC)n1)C(C)C)NC(C(CC)F)=O C(CCCCC(=O)NCC1(C)CCN(C(=O)CN2CCC(C)C2)CC1)OCC C1(CNC(=O)NC2CC(=O)N(C3CCCC3)C2)CNCCC12CCOC2 C(CN=C(NCC1CCC1)N1CCC(N(C)C)CC1)c1c(OC)ccc(Cl)c1 C12(CSC)COC(C(=O)NC(C)CCNC(C3CC3c3n[nH]c(C)n3)=O)(C1)C2 c1(OC)ccc(C(N2CC3C(NC(=O)C(C(C)C)OC)C3C2)=O)c(C(F)(F)F)c1 c1(C(C)(F)F)cc(C(=O)NCCCNC(C2CSCCS2)=O)ccn1 c1(C(C)OCC2CCOC2)nc(-c2ccco2)nn1CC1CCOCC1 N1(C(C2CN(COCc3ccn(CC#C)c3)C(=O)C2)=O)CCC(F)(F)CC1 N1(C(c2nc(C)sc2)=O)CCCC(C)(CNC(C2(N3CCOCC3)CCCC2)=O)C1 C1(C(=O)NCc2cn(C3CCN(C(=O)CCC4CCC4)C3)nn2)(OC)CCSCC1 C(=O)(C(O)C(C)(C)C)NCCN(C(=O)CC1CC1)C(C)C c1(-c2n(C(COCC)C3CC3)ccn2)ccc(C(N)=O)cc1 C(C1=CCCN(C(=O)C(C)c2cc[nH]n2)C1)NC(C(C)CN(C)C)=O N1(C(CCCCCOC)=O)CCC2C(C1)CN2C(=O)C(F)CC1CCOCC1 N1(C(C2(CC)CN(C(=O)CCc3ccsc3)C2)=O)CCC(COC)CC1C c1(C(=O)NCCN(C)C(C2CC2C(F)(F)F)=O)ccc(S(N)(=O)=O)cc1N N1(C(c2c(C)nc[nH]2)=O)CCC(C(N2CCC(Cc3cccs3)CC2)=O)CC1 N1(C(c2cncc(C)c2Cl)=O)CC2CC(NC(c3cnsc3)=O)CC(C2)C1 c1(C(=O)NCCN(C(C2CN3CCC2C3)=O)CC)ccc(C)c(S(N)(=O)=O)c1 CC(C)(C)C#CC(=O)N1CCC(C(C)(C)NC(c2cncc(C(C)(C)C)c2)=O)C1 C(CCCCCCC)NC(=O)CN(C)C(C1CN(C(C(CC=CCC)C)=O)C1)=O Cc1ccc(CN2CCC(C(=O)Nc3cncc(CO)c3)CC2)cc1F N1(C(C(CN(CC)CC)F)=O)CCCC(C)C1CNC(c1cnc(F)c(F)c1)=O N1(C(C23CC(COC)(OC2)C3)=O)CCCC(NC(C2CCC(F)(F)CC2)=O)CC1 C(CCC(C)NC(C1(NC(C2CC3CC3C2)=O)CCC1)=O)OCC N1(C(C(CC)OC)=O)CCN(C(=O)COc2cccc(F)c2F)CC1CCOC C1(CC(=O)O)CN(C(=O)CN2CCCC2c2cccc(Cl)c2)CCO1 CC1(C)C(NC(=O)CCN2CCCC2)CCN1C(C1CCC(=O)O1)=O C1(=O)CCC(C)O1.c12cn(nn1)c(=O)[nH]2.C1(COC)(CO)CCC1 CCC(C)(F)C(=O)NCCc1ccc(CNC(=O)C(C)OC2CCOC2)cc1 c1(C(=O)NCCN2CCC(NC(=O)CCC3CC3)CC2)ccc(F)c(Cl)c1 C1(COC)(NC(=O)CCCSc2ccc(C)cc2)CCN(C(=O)CC(C)O)C1 N1(C(c2nc3onc(C)c3cc2)=O)CC2(CCCCN(C(=O)CNC=O)C2)C1 c1(C(=O)OC(C)(C)C)ccc(C(=O)NCC2CC2NC(c2ccnn2CF)=O)[nH]1 C1(NC(C(CC)=CC)=O)CC(F)CN(C(c2ccc(-c3cscn3)cc2)=O)C1 N1(C(C(CC=C)OC)=O)CCCC(O)(CCNC(=O)C(C)CSC)C1 c1(CCC)ccc(CC(=O)N(CC(O)CCNC(=O)CCc2ccon2)CC)cc1 C(=O)(C1=CCC(NC(=O)CC(C)(O)C2CC2)C1)NC(c1onc(C)n1)C N1(C(CCC(=C)Cl)=O)CC2CCCC(CNC(=O)CNS(=O)(=O)NC)C2C1 c1(C(=O)NCC(N2CCCN(C(C(CCC)OC)=O)CC2)=O)ccc2[nH]ccc2n1 c1(NC(C2CCCCC2NC(c2ccncc2F)=O)=O)cccc(CO)c1 C(=O)(CC1=CCOCC1)OCC(CC)Oc1ccccc1Br.C1(=O)C(C)O1 Cc1cncc(CCC(N2CCCC2C2(O)CN(C(=O)COC3CC3)C2)=O)c1 C=CC(CC)CC(=O)NC1CC2(C1)CC(NC(C1C(C(C)=O)C1(C)C)=O)C2 Cc1cc(C(=O)NCC2CCN(C(=O)CC3CCCC(O)C3)CC2)[nH]c1C CO[Si](C)(C)CCNC(c1ccc(-c2cccs2)o1)=O C1(C)(CNC(C(CC(C)C)C)=O)CC(F)(F)CN1C(=O)CCC1CCC1 c1(CC)ccc(C(=O)N(C)CC2(O)CCN(C(=O)CC3C(C)C3(F)F)C2)cc1 C(=O)(C(O)CCCNC(C1CC(F)C1)=O)NCCCS(C)=O N1(C(C2CC(C)(C)C2)=O)CCC2(CC1)CC2C(=O)NCc1nnnn1C1CC1 C12(NC(C(CC)CC)=O)CCCN(C(c3cc(F)ccc3Br)=O)C1C2 N1(C(C(C)(C)O)=O)CCC2(CCC(NC(=O)CCC3CCCC(=O)N3)CC2)C1 C12(NC(C(C3CC3)OCC)=O)COC(C1)C(NC(=O)Cc1cc(Cl)cnc1C)C2 C(=O)(C#CC1CCOC1)NC(CC=C)C(=O)N1CCC(F)(C(N)=O)C1 c1(C(=O)NCC2N(C(CC3ON=C(CC)C3)=O)CC(O)C2)cc2c(C)cccc2o1 C1(NC(c2n(CC#C)cnn2)=O)CN(C(=O)CCc2nncn2C)CCC1C C1(C(N2CCC(O)(CNC(c3c(CC)nn[nH]3)=O)C2)=O)CCCC2(CCC2)C1 c1(CNC2CC(COC)C2)ccc(OC)c(F)c1F.c12cc(C)c(cn1)[nH]c2=O c1(C(=O)NC(C2C(C(=O)Nc3ncc(OC)nc3)C2)C)c[nH]c2ccccc12 C(c1ccc(Cl)nc1)=CC(=O)NC1(C)CCN(C(c2nccc(N(C)C)c2)=O)C1 CC1CCCC(COC(=O)CCNC2CCN(CNS(C)(=O)=O)CC2)CC1 c1(C(N2C(CNC(CCc3n[nH]c(=N)s3)=O)CCC2)=O)ccc(O)nn1 C1(NC(c2cc(C)nnc2)=O)C2CCC1N(C(c1ccc(=O)n(C)c1)=O)C2 c1(C(N(C2CCN(C(COCCC=C)=O)C2)C)=O)cc(C)c(CC)nc1O C(=O)(C(O)CC(N)=O)N1C2C(NC(CC3(C)CCCCC3)=O)C(C2)C1 N1(C(c2nc(C(C)C)sc2)=O)CCC(C)C(NC(c2ccc(F)cc2)=O)C1 N1(C(c2cnc(OC)nc2C)=O)CCC2CN(C(C3CC(SC)C3)=O)CCC12 CCCCCCC(=O)N1CCN(C(C23CC2COC3(C)C)=O)C(C(C)C)C1 c1(NC(C2(CC)CCCO2)=O)cccc(NC(c2cc(F)n(C)n2)=O)c1 Cc1ccn2ncc(C(=O)NCC34CC3CN(C(=O)CC3CC3(C)C)C4)c2c1 c1(C(=O)NC2CN(C(C(COC)C)=O)CC(NC(C)=O)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC2N(C(COC3(C)CCC3)=O)CC2)cnnn1CCO c1(C(N(C(c2ccccc2)CNC(C(C)CF)=O)C)=O)cc2ccsc2s1 c1(C(N2CCC(NC(CC(C)F)=O)C2C(C)(C)C)=O)ccc2c(c1)OC(C)(C)O2 C12(CNC(C(N3CCC(C)C3)=O)=O)CCC(CC1)N(C(=O)CNC(N)=O)C2 S(=O)(=O)(c1cc(C)ccc1C)NCC(=O)NCCN(C(CC1C(OC)CC1)=O)C C1(CC#C)N(C(=O)C(C)N(C(=O)CNC(=O)CC)CC=C)CCCC1(C)C c1(C(=O)NC2CC3CC(NC(C(CCC)OC)=O)C2C3)nccc2[nH]ccc12 N1(C(C(C)CO)=O)CCC(C)(CCNC(=O)Cc2ccc(Br)cc2)C1 C1(OC(c2ncccc2OCCF)=O)CS(=O)(=O)CC1O CC(C)CC(O)C(=O)NC1CN(C(=O)CCC2CCC(=O)N2)CCC1C Cc1nc2ccc(C(=O)NC(C)(C)CNC(=O)CC3CCNC(=O)C3)cn2n1 C1(F)(C(N2CCC(CN(C(c3c(CC)cncc3)=O)C)C2)=O)CCC(C)CC1 c1(OC)nccc(C(N2CCC(NC(c3ccoc3C)=O)C(F)C2)=O)c1F C(=O)(C(C)C(C)C(C)(C)C)NCCC1CN(C(CCc2c(C)n(C)nc2)=O)C1 c1(CC)ccc(CN2CCCC(C(=O)NC3CONC3=O)C2)cn1 C(=O)(CCCN=[N+]=[N-])NC1(C(N2C(COC)(CO)CCC2)=O)CC1(C)C.C(C)(=O)O c1(C(N2CC(C(=O)Nc3c(C)ccc(Cl)c3)C2)=O)ccnc2c1CC(=O)N2 N1(C(C=CC(CC)C)=O)CC(CNC(c2cnccc2C)=O)C2(CCOCC2)C1 c1(CC(=O)N(C2CCN(C(C3CCNC3=O)=O)C2)CC)ccc2sccc2c1 c1(CN2CCN(Cc3ccc(OCC#C)cc3)CC2)cc(Cl)c(OC)cc1Cl C1(CCC)CN(C(=O)C2=CCCC2)CCN1C(=O)Cc1csc(S)n1 N#Cc1cc(S(=O)(=O)NCC(Cl)Cl)ccc1NC1COc2c(Cl)cccc21 c1(OC)cc(C(=O)NC2CCN(C(=O)CC3CC3C)CC2)c(C)c(Br)c1 C(C1CCN(C(C2C3COCC23)=O)CC1)=CC(=O)N(C1CC1)CC1CC=CCC1 CCC(C)CCCC(=O)N1CC2(CCCC2)C1C(=O)NCC12CCCN1CCC2 N1(C(C(C)(C)OC)=O)CCC(NC(=O)C(c2ccccc2)C)C(CO)CC1 N1(C(CNC(=O)NC)=O)CC(C)(C(=O)N(C2CCC2)CCOC)CC1(C)C Cc1cc(C(c2nnnn2CCCF)NCc2cc(Cl)cc(Cl)c2)cc(C)c1Cl c1(CNC(C)=O)ccc(C(=O)N(C)CCOCCNC(=O)CC2OCCC2C)o1 C1(C(=O)NCC(C)N(C(=O)C(F)CC2CCCC2)C)CCCN(S(C)(=O)=O)C1 Cc1ccc(C(=O)N(C)CC2(O)CCCN(C(C3CCC(F)CC3)=O)C2)cc1Cl c1(CCC)ccc(N)c(C(N2CCCC(N(C)C(C3(O)CCCC3)=O)C2)=O)c1 c1(CNC(CC2CCC(C)C2)=O)ccc(CCNC(=O)C(C)(C)CC2CC2)cc1 Fc1cc(N2CCCC(CCn3nnc(-c4cccs4)n3)C2)cc(F)c1F C12CCN(CC1)C2c1cccnc1.C(C(=O)N(CC(C)NC(C1COC1)=O)C)OC C1(C(C)NC(CN(CCC)C)=O)CCN(C(=O)C(O)CF)CC1 Cc1cnc(C)c(NC(=O)C(=O)NCc2ccccc2Sc2ccncc2)c1 CCC(C)C(C(=O)N(CCNC(c1sncc1C)=O)CC1CC1)c1ccccc1 C1(C(=O)NCCCCCNC(CCc2cc(C)no2)=O)CCC(S(N)(=O)=O)CC1 Cc1cc(C(=O)NC2CC(C)(NC(=O)CNC(N3CCCC3)=O)C2)nn1CCO CC1(C)Oc2cccc(Oc3ccc4c(c3)CN(C(=O)CN)CCCC4)c2O1 N1(Cc2ccc(C)s2)CC(C2CCCN(C(c3cn(C)nc3C)=O)C2)C1 N1(C(c2c(C)nn[nH]2)=O)CCC(C(F)(F)F)C(NC(c2oc(CO)cc2C)=O)C1 N1(CCCC)CC2CCC(NC(=O)CCc3c(C)noc3C)CC2C1 CC(C(=O)NCC(CC(F)(F)F)NC(c1cc2n(c1)CCSC2)=O)C(F)(F)C(F)F CC1(C2CCCN(C(=O)COc3cccc(-c4nnco4)c3)C2)COC(=O)N1 c1(C(=O)NC(c2ccccc2Cc2nn[nH]n2)C)cccc(C(C)(C)C)c1 C(=O)(C1CCOc2ccccc21)NCC1N(C(C(C)SC)=O)CCCC1(C)C CCCC(C=O)C(=O)NCC1CCC1NC(C1(C)CC1)=O.c1(C2CC2)cccs1 c1(C(=O)NCC(C)NC(=O)CC2CCCCO2)ncccc1C(F)(F)F Cc1noc(C)c1CC(=O)NCCC1CC(NC(=O)C(c2ccc(Cl)cc2)C)C1 c1(OC)ccccc1C(=O)NC1CC(NC(=O)Cc2c(C)noc2Cl)C(O)C1 N1(C(C=CCN(C(=O)CC2CSCCO2)C)=O)CCCC1C1(C)CC1 N1(C(C(CC)(C)O)=O)CCC(NC(=O)Cc2cccc(F)c2O)C(CO)C1 C12(CC)COC(C(=O)NCC3(O)CN(C(=O)C(CC)Sc4ccccc4)C3)(C1)C2 C(=O)(C1=CCC(C)CC1)NC1CCC(O)C(O)C1.C12(C(=O)OC)CN(C1)C2=O C1(NC(=O)CC2OCCCO2)CCN(C(C2(c3cccs3)CC2)=O)C1C(C)(C)C c1(C(C(N2CCCC(NC(c3c(CC)occ3)=O)C2)=O)=O)cc(F)cc(Cl)c1 c1(CC(=O)OCC(CCC(=O)NC(C)(C)C)=O)cn2ccsc2n1 Cc1oc(C(C)C)cc1C(N1CC(CNC(=O)CC2OCCO2)C2CC12)=O C12(COC)CC(C(=O)NCC3(OC)CCN(C(c4ccsc4)=O)C3)(CO1)C2 CCC(O)C(=O)NC(C(=O)NC(c1nncn1C)C)c1ccco1 C1(C(=O)NCCC)CN(C(=O)CSc2ccc(C3CCC3)cc2)CC(F)(F)C1 C1(CF)CCCN1Cc1ccc(-c2ccccn2)o1 N1(C(COCCCOC)=O)CCCC1C1CCCN1C(c1cnc(CC)cn1)=O N1(C(c2ccc(C(C)C)cn2)=O)CCC2(CCCCC2NC(C2CCCS2)=O)C1 N1(C(c2ccnn2C2CCCCC2)C(=O)NCCCC)CCOCC1CCOC c1(OC)ncc(Cl)c(C(N2CCC(NC(C3CCCC3(C)C)=O)CC2)=O)c1Cl CC1CCN(C(=O)COc2ccsc2)CC1CNC(c1ncn(C)n1)=O c1(CC(C(=O)N(CCN(C(C=C2CCC(C)C2)=O)C)C)=O)cccc(Cl)c1 C1(COC)(NC(C2CNC(=O)C2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1 S(=O)(=O)(c1cnc(NC2CC2)c(Cl)c1)N1CCC(C(C(N)=O)F)CC1 O=C(C1CCCn2c(O)nnc21)NCc1cn(Cc2cccc(O)c2)nn1 C1(NC(C2CCN(C(C)=O)C2)=O)CC2CN(C(c3cc4n(n3)CCC4)=O)CC2C1 Cc1nccc(C(=O)NCC(C)(C)CC2CN(C(C3CC34CC4)=O)C2)c1C C1(C(=O)OCc2oc(C(=O)OC)c(C)n2)CCC(c2ccccc2)N1CC c1(NC(c2ccc(C(=O)Nc3c(F)cccc3I)[nH]2)=O)c(F)ccc(Cl)c1F c1(C(N2CCC3(CC(NC(C45CSCC4C5)=O)C3)C2)=O)cnc2cccnn12 Cc1nc(C)c(C(N2CCC(CO)(NC(=O)CCC3(O)CCC3)CC2)=O)nc1C C(CC(CO)C(C)C)NC(C(C1N(C(CC2C(CC)C2)=O)CCC1)(C)C)=O.CC Cc1nc2c([nH]1)C(C(=O)NC1CCCC1NC(=O)CN(C)CCO)CCC2 C1(NC(=O)CC2CCOC2)CCN(C(=O)C2=CCCC2)CC12CCC2 N1(C(CN(CC#C)C(c2ccc(C=C)cc2)=O)=O)CC2CC(C1)C2(C)C c1(C(N2CCCC(CNC(CSCC)=O)C2)=O)cc2ccccn2c1 N1(C(CNC(CNC(C)=O)=O)=O)C2CCC1CN(C(=O)Cc1ccsc1Cl)C2 C1(NC(c2c(C)ccnc2)=O)CCCCN(Cc2nc(C(C)(C)C)n[nH]2)C1 C1(CNC(c2cccc(C)c2)=O)CCCC2CN(C(=O)CC3CCCO3)CC12 N1(CC(=O)NC2C(CNC(Cn3c(C)ccc3C)=O)C2)CCN(C)C(=O)C1C c1(C(=O)NCC2(F)CC(NC(C(C=C=C)C)=O)C2)cccc(CC)c1F N1(C(C(CNC(c2c(CC)nns2)=O)F)=O)CC2(C1)CC(C)(F)C2 N1(C(C2(C)CCC(C)CC2)=O)CC2=C(C1)CN(C(c1[nH]nc3ncccc13)=O)C2 C1(O)(c2n(C)ncc2Cl)CCC(C)(C)C1 N1(C(c2nc(C)sc2)=O)CC2CC2(C(N2CCOCC2CCO)=O)C1 C1(N(C)C(c2cnn(-c3ccccc3)c2Cl)=O)CCCN(Cc2cncs2)C1 N1(C(CC(C(F)(F)F)NC(C(CC)(C)C)=O)=O)CC2CCC1C(O)C2O c1(-c2cn(C(C)C(=O)N(CCCn3cc(Cl)cn3)C)nn2)ccc(S(C)=O)cc1 c1(C(=O)NC(CN(C(c2cnc(C)cn2)=O)CC)C)cncc(-n2ccnn2)c1 N1(C(c2scc(OC)c2OC)=O)CC2COCCC2(NC(c2cnco2)=O)C1 C1(NC(C(C#C)(C)C)=O)CCC2CN(C(=O)CC(O)c3ccccc3)CC2C1 C1(NC(=O)Cc2cccc3ncccc23)CCC2CN(C(=O)C=C3CC3)CC2C1 c1(CN2CCCC(C(=O)Nc3c(C(N)=O)cccc3F)C2)c(O)cc(Br)cc1F C(=O)(C(C)C(C)(C)C)NCC(CCNC(CCCOC(C)C)=O)O C1(NC(c2cccc(O)c2Cl)=O)CC2(CCN(C(=O)CC3CC34CC4)CC2)C1 C(=O)(C(O)CC(C)(C)C)NCC(CNC(c1cccc(OC)c1C)=O)O Cc1cc(F)c(C(=O)NCC2CN(C(=O)C(C)N3CCC3)CC2(F)F)c(F)c1 C1(NC(Cc2scc(C)c2)=O)CC(O)CN(C(=O)CN(c2ccc(Cl)cc2)C)C1 C1(C(=O)NCC2(CN(C)C(C3CC3(C)C)=O)CC2)CCC(=O)C1 c1(C(=O)OC)ccc(Br)c2[nH]nc(C(N3CCCC4(CCC4)C3C)=O)c12 c1(OC)cccc(Br)c1C(N1C2CCC(C2)C1C(N1CCOC(=O)C1)=O)=O C1(CC(=O)NC2CN(C(CCSC3(C)CC3)=O)CC2C(F)F)CCCC(F)(F)C1 C1(NC(c2csc(Br)c2)=O)CC(=O)N(C2CN(CC(O)Cn3cccn3)C2)C1 CC(C)(C#N)CCCC(=O)NCCCC(O)C(=O)NCc1cc(C2CC2)on1 C1(CCNC(CC(C)OC)=O)CN(C(=O)CCCC(N)=O)CCS1(=O)=O c1(-n2cc(C(C)(C)NC(c3c(COC)oc(C)c3)=O)nn2)cnc(F)c(F)c1 Cc1ccc(C)c(C(=O)NC2CCOCC2C(=O)NC(c2ccco2)CO)n1 CCC(C(=O)N1CCC(C)C1CNC(c1cc(O)nc(O)n1)=O)C(C)O C(CC(F)F)(C(=O)NCC(C)(O)CN(C)C)N(C(CC(CC)C1CC1)=O)C Cn1nc(C(=O)NCC2(F)CN(C(=O)CC3CCNC(=O)C3)C2)cc1C1CC1 N1(C(C=CCOCCOC)=O)CCCC12CCN(C(=O)CS(=O)(=O)C(C)(C)C)C2 C1(CC(=O)NC2CC2NC(c2ccc([N+](=O)[O-])cc2)=O)CCC2(CCC2)CO1 n1(CCCC)[nH]c(=NC(=O)C(F)(F)C(O)C(C)C)cc1C#N c1(CNC2CCC(C(=O)Nc3c(C)[nH]nc3Cl)C2)cc2cnccc2[nH]1 c1(OC)c(C(N2CCN(C(=O)CC3CC3)CC2CC2CC2)=O)c(C)nn1C C1(CNC(c2ccn(C)c2)=O)CN(C(c2cccnc2F)=O)CCC12CCC2 C(=O)(C1=C(Cl)CCC1)NCC12CC(NC(c3c(C)n(C(C)C)nc3)=O)(C1)C2 CCCC(C)CCNC(C1CC(CCNC(=O)CCC2CC2(C)C)C1)=O CC(C(=O)NCC(C1CC1)NC(c1cnc(-c2ccccc2)[nH]1)=O)C(C)(F)F c1(C(=O)NCC23C(NC(c4c(C)nn[nH]4)=O)CC(CC2)C3)ccn2c1CCCC2 CC(C)(C)C1=NOC(C(=O)NCCCCCNC(C2CCS2(=O)=O)=O)C1 c1(C(N2CCCC(F)(CNC(C3(C)CCC3)=O)C2)=O)ccc2c(c1)NCCO2 C1(NC(C(c2cncnc2)C)=O)CC(=O)N(C2CN(C(=O)C(F)=CC3CC3)C2)C1 N1(C(CCC=C)=O)CCN(C(c2cc(OC)c(Cl)cc2Cl)=O)C(C)C1C c1(OCCCC(=O)NC2(C)CC(NC(C(CC)(C)C)=O)C2)ccc(C)c(C)c1 c1(C(=O)NCC(CC(F)(F)F)NC(C2(OC)CCSC2)=O)ccnc2cc[nH]c12 c1(NC(C)=O)ccc(Cl)c(C(=O)NCCNC2CCC2F)c1 N1(C(C2CC(C)SCC2)=O)CCC2(CCCN2C(=O)CNC=O)C1 CC(CC(=O)NC(CCC1CC1)C(=O)NC1(c2cc[nH]n2)CC1)C(F)F N1(CCN(C)C(c2ccn(C3CC3)c2)=O)CCC(NC(C2CSC2)=O)CC1 c1(NC(=O)NCC2N(C(CC3C(C(=O)OCC)C3)=O)CCC2)ccccc1Cl N1(C(C)=O)CCCC(C2CCN(C(C3(N(C)C)CC3)=O)C2)C1.CCC(C)SC c1(COC)cc(O)nc(NC(=O)C(C)NC(=O)CCOCCN)n1.SC c1(C(=O)NC(C2(CNC(c3cc(CCC)on3)=O)CC2)C)nc(C)sc1C c1(C(=O)NCC2CN(C(CC(=O)NC3CC3)=O)CC2O)cnn2ncccc12 C1(C(N2C(CONC(c3cc(C4CC4)on3)=O)CC2)=O)C2CCCCCC12 C1(C)CN=C2C=C(N=C(C(C)C)N2)C(=O)N1.c1(CC)ccnc(COC)c1 c1(OC)cc(CCNC(=O)CCC2CCCNC2)cc(OC)c1OC c1(C(c2nnnn2Cc2ccco2)NCC2C=CC(OC)C2)c(C)ncnc1C CCCC(CCNC(C1CCN(C(=O)COC)C1)=O)C1CC1 CCCC(C)CC(=O)N1CCC(N2CC(C)(CNC(C3CCSC3)=O)C2=O)CC1 C#CC1(CC)COCCN1CC(=O)Nc1cccc(Cl)c1Cl c1(C(=O)NC(C(C)NC(C=Cc2n(CC)ncc2)=O)C)ncc(F)cc1F N1(C(c2c(C)nc(OC)s2)=O)CC2CN(C(c3cc(C)n(C)n3)=O)CCC12 N1(C(C(CC2CC2)OC)=O)Cc2[nH]nc(C(=O)NC3C(C)CCC3C)c2C1 Cc1cc(Cl)ccc1N(CCC#N)C(N1CCN(c2nccn2C)CC1)=O C12(C(N3CC(N(C(c4ccnc(OC)n4)=O)C)C3)=O)CCC(C)(C(=O)O1)C2(C)C CCC(C)(COC)C(=O)NCCC1CCN1C(=O)CC=C(C)C.c1(CC)ccccc1 CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCC1CNC(=O)C(C)(C)C#N C1(NC(C(c2cncn2C)N(C)C)=O)CCN(C(c2n[nH]c3c2COC3)=O)C1(C)C CCC(C(=O)N1CCC(CC(=O)NCCN(C)CCOC)C1)C(C)(C)CC c1(C(=O)NCC2C(NC(C(F)=C(C)C)=O)CC2)cccc(F)c1Br N1(C(C(C)NC(c2cscc2Cl)=O)=O)CCC(C2CCC2)CC1 N1(C(C2CCCN(Cc3ccc(OC)cc3)C2)=O)CCC2(CC1)CN(C)C2 c1(C(=O)NC2CCCC(NC(=O)CSC(F)F)C2)ccc(Cl)c2cccnc12 C1(NC(=O)C=CC2CCCO2)(CO)CN(C(=O)COC(F)F)C1 c1(CNC(c2ccc(C(F)(F)F)cc2)C(=O)OC)ccccc1-c1ccccc1 c1(CC(C)C)nc(Br)cnc1NCc1ccccc1OC1COC1 N1(C(CCCCC(=O)OC)=O)CC(C2CCCN(C(c3nc[nH]n3)=O)C2)C1 C1(COC)(NC(C2C=CCN2C(C23COCC2C3)=O)=O)CCCCC1 c1(C(N(C2CCN(C(C(CCC)OC)=O)C2)CC)=O)ccc(Cl)cc1Cl c1(N(C(C)C)C)nnc(-c2ccccc2Cl)n1CCCN1CCOCC1 CN1CCCC2CN(S(=O)(=O)C3CC(N)C3)CCC12 N1(C(CCNC(C)=O)=O)CCC(O)(CNC(=O)CC2CC2c2ccccc2Cl)C1 CC1(C)C(CNC(C2CC2C2CC2)=O)CCN1C(=O)CCN1CCCCC1=O O=C(C1=NOC2(CCOC2)C1)NC1CCCC12CN(C(=O)C=CI)C2 c1(C(=O)OC)cc(C(=O)NCC2CCCN2C(C2CC(C(N)=O)C2)=O)cc(Br)c1 N1(C(N(C2CCC(C(=O)OC)CC2)C)=O)CC(CO)CC(CO)C1 C1(NC(N2CCCC(C(C)(C)O)C2)=O)CCc2nnsc2C1 N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCC(OC(=O)N(C)Cc2ccc(Cl)nc2)CC1 c1(C(=O)NCC2C(C)(C)CN(C(c3cc(Cl)no3)=O)C2)ccc([N+](=O)[O-])cc1 C1(NC(CC(CC)C)=O)CCCC(N=c2[nH]c3c(F)cccc3o2)C1 c1(OC)cc(C)c(CNC(=O)N(C)Cc2ccoc2C)cc1OC CC1=C(C)CC(C(=O)NCCCN(C(=O)Cn2ncc(O)nc2=O)C2CC2)CC1 C(=O)(C1OC(=O)c2ccccc21)NC(CN(C(c1ccc(OC)cc1)=O)CC)C C(=O)(C#CC1(C)CCCO1)N(C(C)C(=O)NCC(=C1CCCCC1)F)C1CC1 C(=O)(CCCCC(=O)NCCCN(C(=O)C(C)(F)F)CCO)NC c1(C(N(CCN(C(c2cc(C(=O)OC)sc2)=O)C)C)=O)c(C)c[nH]c1CC(N)=O c1(C(=O)NC2CCN(C(C(C)(C)OCC)=O)CC2O)cccc2nn[nH]c12 c1(C(N(CC(=O)NC(c2n(C)ncc2)CO)C2CCC2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(C2(CCC=C)CC2)=O)CC2(CCC(CNC(=O)CCc3ccccc3)O2)C1 Cc1cccc2oc(=NCCCNCc3cnn(CC4CCCC4)c3)[nH]c12 c1(OC)ncc(Cl)c(C(=O)NCC(C)N(C)C(c2c(C)nn(C)c2Cl)=O)c1Cl c1(C(=O)NC(c2cc(C)no2)C)cc(C)c(-c2cccs2)s1 N1(C(C(C)NC(CC)(C)C)=O)CC2(CCN(C(=O)C3=NOCC3)CC2)C1 C(=O)(CP(C)(C)=O)N(CC(NOC(=O)C(C)C(C)C)=O)CC C(C(CNC(=O)Cc1ccsn1)CO)NC(C1CC(SC)C1)=O N1(C(C(CC=C)CC)=O)CCCC2(CCCN2C(=O)C=CC2(C)COC2)C1 C(=O)(CP(C)(C)=O)NC(C1CCCC1)CNC(c1c(CC(=O)OCC)scc1)=O N1(C(C)=O)CCC2(CC1)CC(NC(c1nn(C(C)C)cc1Br)=O)C2 CN1CCCC(C(=O)NCCCC2(NC(=O)CCc3cccnc3Cl)CC2)C1 c1(CNC(c2cnc(C)s2)=O)cccc(C(N2CCCC(C(=O)N(C)C)C2)=O)n1 C1(NC(C(C)OC2CCCCCC2)=O)CC2CCC(C1C)N2C(=O)CC1CC1C c1(-c2ccc(C)c(F)c2)ccn2ncc(C(=O)Nc3cc(Cl)cc(F)c3I)c2c1 N1(C(CCC)=O)CC2(C1)CN(C(=O)C#CC1CCOC1)CCO2 CCC(C)S(=O)(=O)C(C(=O)C(=O)OC(C)(C)C)c1nc2ccc(C)cc2s1 C1(NC(c2ccc(C)cn2)=O)CCCC12CN(C(C1CC3C(C1)C3(F)F)=O)C2 c1(CNC(=O)CC2CSC2)conc1C(N1CC(O)C1)=O C(CCC)(C(O)C(=O)N1CC(C)(CCOC)C1)NC(C(C=C)O)=O C1(CNC(c2cc(C3CC3)ccn2)=O)CN(C(=O)C#CC2CC2)CCO1 C1(C)(OC)CN(CC(=O)NC2CC(C(=O)NCC(c3ncc(C)s3)C)C2)C1 C1(C(=O)NC(CC)CNC(c2nc(C)nn2C)=O)CC2CC(OC)C2C1 Cc1cc2[nH]c(=O)c(C(N3CCC(CNC(c4n[nH]c(C)c4Cl)=O)C3)=O)cn2n1 CC1CN(C(=O)C#CC(C)(C)O)CCN1C(C1CCOC(C)(C)C1)=O c1(OC)ccc(C(=O)NC2CC2C(=O)Nc2nccnc2Br)c(Cl)c1OC c1(OC)ccc(F)c(C(=O)NC2CCN(C(=O)Cc3cn[nH]c3)CC2CO)c1F Cc1cn2cc(C(=O)NCC3CCN(C(=O)Cc4cn[nH]c4)CC3C)sc2n1 C1(NC(C(C)OCC)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CCC1(F)F CCC(C(=O)N1CCCOC(CCNC(c2cccc(CO)c2)=O)C1)C(C)(F)F Cn1ccc(O)nc1=NC(=O)N1CCCC1c1ccc(Br)s1 c1(C(=O)NCC2CCN2C(=O)C(O)C2CCC2)occ2c1CCCC2 C(=O)(CCCCC(C)(C)C)N1C(C(=O)NCC(CC)N(C)C)CC=CC1 C1(C(=O)NCC2N(C(=O)Cc3cn[nH]c3)CCCCC2)CC(F)(F)C12CCC2 C=CCCC(=O)NCCC1(NC(=O)CCc2nc(SCc3ccsc3)no2)CC1 c1(C(C)=O)ccc(C(N2CCC(C)C(NC(=O)C(O)C3CC3)C2)=O)c(F)c1 Cc1ccc2nc(CC(N3CCC(C)C3CNC(=O)C#CC3(C)CC3)=O)[nH]c2c1 c1(CC)nc(N2CCN(C(C3CCCSC3C)=O)CC2)cc(C#N)n1 C1(NC(CS(C)(=O)=O)=O)COC2CN(C(=O)CCCCc3ccccc3)CC12 C(CCCC(=O)NCC1CCCN(C(=O)Cc2csc(Cl)c2)C1)N(C)C N1(C(C=C(CC)CC)=O)CCCC(C)(C)C1CNC(C1C(C)C1(F)F)=O n1(CC(N2CCC(NC(Cc3nnc(C)o3)=O)C2)=O)ncc(C#N)c1Br N1(Cc2ccc(C(=O)OC)o2)CCC2(CCN(C(c3ccc(Br)s3)=O)C2)C1 C1(C(=O)NCC2(C(=O)NCC(c3cncs3)O)CC2)CCCN1C1CC1 Cc1ccncc1CC(=O)NCCCOC1CCN(C(=O)CC2CCCO2)CC1 C1(C(=O)NCCCCn2ccnc2)CC=CCN1C(=O)CN1CCCC1=O N1(C(c2ncn(CCNC(C(C)C(F)(F)F)=O)c2)=O)CCCC2COCC12 CC1CN(C(C2CC2(C)C)=O)CC1NC(=O)CSCc1cccnc1 C(C(C)(CC(C)C)NC(c1cnc(C2CC2)s1)=O)NC(CCC=CCC=C)=O CC#CCCC(=O)NC(C1(O)CCN(C(c2oc(C)nc2C(F)(F)F)=O)C1)C C1(CC(=O)NC2CCC(CNC(=O)CC3(O)COC3)C2)CC2CCC1O2 C1(C(N2CCC(NC(c3cnc(C)s3)=O)C2)=O)CC(=O)N(CC(F)(F)F)C1 Cc1c(Cl)nc[nH]c1=NCC1(CNC(=O)CN2CCS(=O)(=O)CC2)COC1 N1(C(C(C(C)C)NC=O)=O)CCC(C2CN(C(=O)COCC(C)(C)C)C2)C1 c1(C(=O)OCC)ccccc1CN(C(C)C(=O)NCC(C1CCCO1)=O)C c1(NCC)cnn(C2CCN(C(c3nc(C4CC4)cs3)C)CC2)c1C C1(NC(CSCC)=O)CCCCC12CCN(C(c1cc3n(c1)CCCC3)=O)CC2 C1(CNC(C=COCC)=O)CCN(C(c2ccc(C(N)=O)nc2)=O)C1(C)C C1(C(=O)NCC=CCNC(c2cocn2)=O)CCCN(c2ccc(Cl)nn2)C1 N1(C(Cc2c(CC)con2)=O)CC2CC(NC(c3n[nH]c(O)n3)=O)C2C1 c1(NC(CCOC)=O)cc(NC(N2C(C(CCCCl)OC)CCC2)=O)ccc1F N1(C(CCNC(C)=O)=O)CCC(C=CC(=O)NC(C)C(C)n2cncn2)CC1 N1(C(C(c2cc(C)c(F)cc2)(C)C)=O)C2CCC1C(C)C(NC(C1CSC1)=O)C2 c1(C(N2CCCN(C(C3C(CC)CCO3)=O)CC2)=O)csc2c1CCCC2 C1(NC(C=C(C)C(F)F)=O)CCN(C(=O)C=CC(c2cnn(C)c2)=O)C1 C1(CC)CC(O)CN1C(C1COCCC1NC(=O)C(C1CC1)C1CC1)=O c1(CN2C(C(=O)Nc3c(CC)nc[nH]3)CC(O)C2)ccc(F)c(C(F)(F)F)c1F C1(OC(C)=O)CCCN(C(C2C3CN(C(C4CCCN4C4CC4)=O)CC23)=O)C1 CC1CC(=O)NC(C(=O)NCCC2(O)CN(C(=O)CSCc3ccccn3)C2)C1 c1(NS(C)(=O)=O)ccc(NC(=O)NC2CC2NC(=O)CC2CCC2)cc1F CC1CN2CCC1NCCC2=O.C1(C(=O)NCC(N)=O)CCCCS1 CC1(C)CNC(=O)N(CC(C)(C#N)c2ccccc2)C1=O.O1NC1 C1(NC(CCC=CC(C)C)=O)CCN(C(=O)CSc2nc[nH]n2)CC1O C1(C(C(=O)N(CCOCCO)CC)(C)C)CCCN(C(=O)CN(C2CCC2)C)C1 C(C(C)N=c1nc[nH]c2[nH]c(Cl)cc12)N(C(C(CC)NC(N)=O)=O)C C1(CCC(=O)N(CCCCN(C)C)CCCCCNC(=O)CO)CC2CCC1C2 C(CCCC(=O)N1CCC(C)(CCNC(=O)C(O)CC2CC2)C1)OCCC=C C(C)(C(=O)N1CCC(CC(=O)NC(C)C(C)(C)O)C1)(C(C)C)NC(C)=O C(=O)(CS(C)(=O)=O)N(CC(C)(C)CNC(=O)C(C1CCCO1)OC)CC Cc1cc(OC(C2CSC(C(F)(F)F)C2)=O)ccc1[N+](=O)[O-] C#CCC(O)C(=O)NC1CN(C(=O)CCCN(C)C(C)=O)CC1F C1(COC)C(NC(c2cn(CC3CC3)nn2)=O)CCN1C(=O)C1=COCC1 N1(C(c2nnn(C)n2)=O)CC2(CCN(C(c3ccc4c(n3)OCCO4)=O)CC2)C1 N1(C(C(CC2CCC2)OC)=O)CCCC(C)(CNC(=O)CN(C(=O)C(C)C)C)C1 C(=O)(C(C(C)C)N1CCN(C)CC1)NC(CC)CNC(=O)CC1(NC(C)=O)CC1 C1(C(N2CC(O)(CCNC(C3C4CCC34)=O)C2)=O)(OCC)CCCCCC1 CCC1=NOC(CC(=O)OC)C1.C12(CN(C(=O)C(C)NC(=O)C(C)(C)C)C1)C(=O)N2 c1(CNC(c2cc(F)ncc2NCc2ccoc2)=O)cc(Cl)cc(Br)c1 C=CCCCCCC(=O)NCC1CCN(C(c2cc(SC)c(Cl)cc2Cl)=O)C1 c1(NC(C(C=C)OC)=O)ccc(NC(=O)CC(C)COC)c(C)c1 C=CC1(CNC(=O)C(N2CCC(SC)C2)=O)CCC1 c1(C(=O)NC2C(NC(=O)Cn3nnc(=O)[nH]3)CC2)ccc([N+](=O)[O-])[nH]1 c1(OC(CC)C(=O)NC(C)(C)CCNC(C2(CO)CCCC2)=O)ccccc1C N1(C(C(C(C)C)=O)=O)CCCC(C2(NC(=O)C=C3CCN(C)CC3)CC2)C1 N1(C(C2CC(NC(C3CCCO3)=O)C2)=O)CCC(Oc2ccccc2Cl)CC1 c1(OCC=C)cccc(Cc2nc(CN3CCCC3)nn2-c2cnnn2C)c1 c1(CC)ccc(C(=O)NC2CC(NC(C3(OC)CS(=O)(=O)C3)=O)C2)cc1F n1(CC(=O)NCCCNC(C2(C)CCOC2)=O)ccc(=O)c([N+](=O)[O-])c1 N=c1[nH]c(N2CCC(CC3CCCC3)C2)nc2ccc(F)cc12 N1(C(C2CCC3(CCC3)CC2)=O)CC2CCCC(C1)N2C(C1CCCC(O)C1)=O c1(C(N2C(CNC(C3OCCN(CC)C3)=O)CC2)=O)cc(F)ccc1N c1(NC(C2C(CNC(=O)C=Cc3cocn3)OCC2)=O)ncnc2[nH]cnc12 c1(C(=O)OCC)ccc(C(=O)OCCN(CC(C)O)C)cc1Br CCCCCCC(CN(C(=O)C(N1CC(F)(c2ccccc2)C1)=O)C)CC c1(OCC(=O)NCC2(NC(COCC)=O)CC2)ccc(O)cc1.c1(O)ccc(O)cc1 Cc1nn(C)c(Cl)c1C(=O)NCC(C)NC(c1coc(C(C)(C)C)n1)=O C1(COC(C=CC)=O)CC12CCS(=O)(=O)CC2 c1(C(N2CCC(CNC(C3(CF)CC3)=O)C2)=O)cc(O)nc(O)c1 N1(C(c2c(C(C)NC(CC(CCC)C)=O)noc2)=O)CCOC(C)(C)CC1 C1(OC)CC(C(=O)NC2CC(NC(c3scnc3C3CC3)=O)C2)C12CCC2 Cc1c(C(=O)NC2CC2NC(=O)CCC(F)(F)F)cccc1F C1(NC(Cc2ccc(OC)cn2)=O)CC2CC(NC(=O)C(C)c3ccsc3)C2C1 c1(C2C(C(=O)NC3CC(CNC(=O)CCF)C3)C2)cccc(Cl)c1 C1(NC(CN(CCC)C)=O)C(C)CCN(C(C2CC=CCC2C)=O)C1C CC1(C)COCCC1CC(N1CCCC(NC(=O)CN2CC3C=CC2C3)CC1)=O c1(C(=O)NC(C2CCN(C(c3cc(C(=O)OC)on3)=O)C2)C)ccccc1O c1(C(=O)NCCC2(NC(COC)=O)CCCC2)ccnc2c1CCC2 N1(C(C(N2CC(C)N(c3nccn3C)CC2)=O)=O)CCC2(CC1)CN(C)C2 C=CCCCC(C)(C)C(=O)NCCCC(N1CCC(C)=C(F)C1)=O C(=O)(C(F)(F)C(O)C1CC1)NC1(CNC(=O)CC(c2ccccc2)C2CC2)CC1 C1(CC)C(C(=O)NCC(C)(C)C#N)CCN1C(=O)C=NOC c1(OC)ccc(C(=O)NC2CC2C(=O)NCC(=O)N(C)C)c(F)c1 c1(N(C(CC(C)OC)=O)C2CCC2)ccc(F)c(F)c1 N1(C(C(C)OCC#C)=O)CC(CO)C2(C1)CN(C(C13CCC(CC1O)C3)=O)C2 C1(C(=O)NCC2CC(C)CN(C(=O)CCCC(F)(F)F)C2)CC2(CCCC2)CO1 Cc1cc(C(N2C(CNC(c3nnc(O)nc3O)=O)CC3CC23)=O)cnc1C c1(C(=O)NC)nc(N2CCC(C)(C)C2CN)c2scc(C)c2n1 CCCCC(O)C(C)C(=O)NCCC1COCCN1C(=O)C(C)=Cn1ccnn1 c1(C(=O)NCC2CC(C)N(C(C3CC(Cl)(Cl)C3)=O)C2)c(F)ccc(Cl)c1F N1(C2CN(C(c3ccccc3)=O)CC2O)CCc2cnc(C3CC3)nc2C1 c1(C(=O)NC2C(CC)CN(C(C)=O)CC2)ccc2c(n1)OCCO2 C1(NC(CCOc2c(C)cccc2)=O)CCN(C(C2(CF)CCC2)=O)CC1C C(=O)(C1=CCSC1)N(C(C)CN(C(=O)C(C)Sc1ccncc1)C)C c1(C(N2CC(CC(CNC(C=C(CC)CC)=O)(C)C)C2)=O)cc2cccc(O)c2[nH]1 c1(OC)ccc(F)cc1C(=O)NC1CC(C)N(C(c2ccc(CO)cn2)=O)C1 C1(CNC(C(C)n2ccnc2)=O)CN(C(=O)CCNS(C)(=O)=O)CC1C c1(C(=O)NC(CNC(c2cccc(NC(=O)OC)c2)=O)C)csc2ccncc12 N1(C(C2(C#C)CC2)=O)CCC(NC(=O)Cc2cncs2)C(CO)C1 N1(C(C2(C)ON=C(C(C)C)C2)=O)CCC2(CCN(C(=O)CCF)C2)C1 N1(C(CC2C(C)(C)OCC2)=O)CCC2(CC2NC(c2cnc(C3CC3)o2)=O)C1 Cc1ccc(O)cc1C(N1CCN(C(c2c(C(F)F)n[nH]c2C)=O)CC1CO)=O C1(CC)CCCN(C(=NCCN(C)C(C)=O)NCC(CC)C(C)C)C1 C1(NC(c2c(C)noc2C)=O)CN(C(=O)C=Cc2ccc(Cl)cc2)CCC1F c1(-c2ccc(CNC(c3ccc(OCC)nn3)=O)nc2)ccc([N+](=O)[O-])c(C)c1 C1(C(C)C)CN(C(=O)CC2CSC2)CCN1C(=O)CC1CCC(=O)N1 c1(CNCc2c(OC)cncc2)c(O)cccc1F C1(NC(CCC#C)=O)CCN(C(=O)COc2c(CC)cccc2CC)CC1CC N1(C(=O)NCC)CC(N=c2[nH]c(=NCCCN3CCOCC3)[nH]c3ncn(C)c23)C1 C(C)(C(C(=O)N1CC(c2cc(O)n[nH]2)C1)NC(=O)C=CC1(C)COC1)OC CCCCCCC(=O)NCc1ncoc1C1CN(C(C2CC(=O)C2(C)C)=O)C1 c1(C(N2CCC(NC(c3cc(COC)no3)=O)C2C)=O)cccn2nccc12 C#Cc1cn(C)nc1C(N1CCC(O)(CCNC(=O)C(C)=CC2CC2)CC1)=O C1(C)(CC)CC(NC(=O)C2CC2)CN1C(c1cc(C2CC2)ccc1F)=O c1(C(N2CCC(NC(CC3CC(OC)C3)=O)C(O)C2)=O)cc(Cl)cc(Cl)c1N C1(C(=O)NC(CC=C)C(=O)NC2CC(C)(C)C23CC3)CC(=O)NC(=O)C1 c1(C(=O)NCCOC2CN(C(c3ccc(F)s3)=O)C2)cc2nc(F)ccc2o1 CN1CCN(S(=O)(=O)N2CCCC(NC(C3CCC(C(=O)O)CC3)=O)C2)CC1 c1(C(=O)NC(CNC(C(CCSC)O)=O)C2CCC2)cc2cccn2c(O)n1 C(=O)(C(C)CC(F)(F)F)NCC(C(=O)NCc1c(C)cccc1)C(C)C C1(C)(NC(CCN(C(C(C=C)OC)=O)C(C)C)=O)CCC(C)(C)C1 N1(C(Cc2ccc(C)s2)=O)CCCC(C(=O)N(C(C)CC(C)C)C)C1C n1(CC)cnc2nc(N3CCC(C)(CO)C3)[nH]c(=NC(C)c3ccc(Br)nc3)c12 C=CC1(CC(=O)NCC(C)N=[N+]=[N-])CN(C(C2CC2CC(C)(C)C)=O)C1 C12(C(=O)NC3CC(CNC(C(C(C)C)OC)=O)CC3O)CC3CC1C2C3O c1(CC(=O)N(CCCNC(=O)CSCc2ccco2)C)cccc(F)c1F C1(C(=O)NCCn2ccnc2)CC2CC2N1C(c1ccccc1)c1sccc1Cl C1(CC)CCC(C(=O)NCC(F)CNC(c2ccc(C(C)=O)cc2)=O)CC1 Cc1c(C(N2CC(CC(F)C(N3CC(C)OCC3C)=O)C2)=O)[nH]ccc1=O N1(C(CN(C(C)C)C(=O)OC(C)(C)C)=O)CCCC(NC(C2CCC2(C)C)=O)C1 C=C1CC(C(=O)NOCCC(C)O)(CNC(=O)C(C)Cn2ccnc2)C1 c1(C(=O)NCC(CO)NC(c2cc(C)[nH]c2C)=O)csc2ccccc12 CC(C(=O)NC1(C(=O)NCc2ccc(F)c(F)c2)CC(O)C1)S(N)(=O)=O C(=O)(C(O)CC(C)(C)C)N1CCN(c2c(OCC(=O)OC)cccc2Cl)CC1 C(C)(C(=O)N1CCC1C(=O)NCc1cccc(F)c1C)(C(C)C)OC c1(C(=O)OC)cc(C(N2CCN(C(=O)CC3(C)CC3)C3CC23)=O)c(F)cn1 C(C)(CCCCNC(c1ccc(C(F)F)s1)=O)NC(CCc1scc(C)n1)=O c1(C(N2C3CC(NC(C(C)=C(C)C)=O)(C3)C2)=O)cc(N(C)C)nc2ccccc12 C1(C(N2CCCC(C3N(CC(C)OC)CCCC3)C2)=O)COc2ccccc2O1 C(C(C)(C)C1=CCOCC1)NC(N(c1nc(CC2CC2c2ccccc2)cs1)C)=O C(=O)(C1=CCCOCC1)NC1CCC(C)(NC(C2CCC(C)(C)OC2)=O)CC1 c1(SC)sccc1C(N1CCCC1C(C)(C)NC(C1(C)CC(F)C1)=O)=O C1(C(=O)NCCC(C)(C)NC(c2cccnc2O)=O)CC2(C1)CC(F)(F)C2 c1(C(=O)NCC2CC(OC)CN2C(=O)CCC(C)O)cc(C)nc(O)n1 Cc1nc2nccc(C(N3CCC(c4cccs4)CC3)=O)n2n1 C(=O)(C(C)(O)C(F)(F)F)NCC(CC(=O)N(CC=C)CCO)O Cc1cc2ncc(-c3ccc(NC(c4cccc(O)c4O)=O)s3)cn2n1 C=CCC(C(=O)NC(C)CCCCNC(C1CN(C(C)=O)C1)=O)OC C=C1CCC(C(=O)NCc2nc(C(=O)NCCC(=O)NCC)co2)CC1 N1(C(C(CC)COC)=O)CC2(CCCN(C(=O)COc3cc(C)on3)C2)C1 C1(C)(NC(C2CCN(CC(C)C)C2)=O)CCN(CCOC2CC2)C1 c1(C(N2C(CNC(c3n(CC)ccc3)=O)CC2)=O)cncc(OCC(F)F)c1 c1(C(=O)NCCc2n(C)ncn2)cc(-c2sccc2Cl)cn2ccnc12 c1(CNC(C(C=CC)O)=O)ccccc1CNC(=O)C(C)OCC C1(CN(C)C(C2CCOC(C)C2)=O)CN(C(c2cccc(C)c2N)=O)CC12CC2 C=CC(CC)CC(=O)NCC(c1cccc(C)c1)NC(c1ccoc1C)=O c1(CC(=O)NCC2CCC2C(N(CC(C)C)CC(C)C)=O)ccc(F)cc1Cl c1(C(N(C2CCN(C(C3CCC(=O)O3)=O)C2)CCC)=O)cc(C(F)(F)F)cn1C c1(C(=O)NCC2(O)CCCN(C(c3cnc(O)o3)=O)C2)ccc2nccnc2c1 N1(C(c2cc(NC(=O)OC(C)(C)C)sc2)=O)Cc2ccccc2C(CO)C1 c1(CCC(=O)NCCC2(NC(C3C(C(=O)OC)CC3)=O)CC2)ccccc1F N1(C(C=CCC)=O)CCCC1C1CCCN1C(=O)C=Cc1c(C)noc1C c1(C(=O)NC2CC(C)(NC(C(CC)N(C)C)=O)C2)cnc2n1CCS2 S(=O)(=O)(c1cc(Cl)ccc1F)N1CCC(C#N)(Nc2ccc3c(c2)CCC3)C1 N1(C(c2ccc(OC)s2)=O)CCC(O)(C2(NC(=O)Cn3ncnn3)CC2)CC1 N1(C(COCCC#C)=O)CCCN(C(=O)CCc2ccc(OC)cc2)C(C)C1 N1(C(C2N(C(=O)OC)CSC2)=O)CCc2sc(CNC(C3C4CCC34)=O)nc2C1 Nc1cc(Cl)ncc1C(=O)NCc1nc(CNC(=O)C2=NOCC2)cs1 N1(C(c2c(NCC)cc(Cl)cc2)=O)CCC2(C1)CN(C(=O)C(C1CCC1)OC)C2 C1(N(C(=O)C=CCF)C)CCN(C(C2CCCN2C(=O)C(C)(C)C)=O)C1 N1(C(CC(=C)C)=O)CCCCC1CN(C)C(C1(CSC)CC1)=O Cc1nc2c(s1)CN(C(c1ccc(CNC(C3(C)CCC(C)C3)=O)cc1)=O)C2 C(=O)(C1=CCC(C(F)(F)F)OC1)N1CC(NC(CN(CC)CC)=O)C(F)C1 c1(C(C)NC(c2ccc(Br)c(C(F)(F)F)c2)C)cccc(O)c1Cl C1(CN(C(CSCCC)=O)C)CN(C(C2CC2(C(C)C)COC)=O)CCO1 n1(CCC)cc(C(=O)NCC2(NC(=O)C(F)C3CCOC3)CC(F)(F)C2)c(C)n1 Cc1cc(=O)n(C)cc1C(N1CC2CCCC2(NC(=O)CCOC2CC2)C1)=O C1(NC(c2cnn(CC)n2)=O)CCCCC1NC(=O)C1CC1.C12CCCN1C2=O CCC(CC(=O)NC(C1CCN(C(C2Cc3ccccc3O2)=O)C1)C)C(C)(C)C c1(Cn2cc(C3(O)CN(C(C4(C)CC4(Cl)Cl)=O)C3)nn2)ccccc1[N+](=O)[O-] c1(C(=O)NC(CN(C(=O)CCCOC)CC)C)n[nH]c(C2CC2)c1Br C(CC(=O)NC1CC(CF)C1)(C(F)F)NC(C1C(OC(C)=O)C1)=O.C1(N)CCOC1 CC1CN(C(=O)Cc2ccc(Cl)s2)CC1NC(=O)CCc1cnc(C2(C)CC2)o1 c1(NC(=O)C)ccc(Br)cc1Cl.N1(C(CC(C)C)=O)CC(N2CCNCC2)C(F)C1 C=C1CC2(C1)CC(C(=O)NC1CC(C)(NC(C3CC3C(F)F)=O)C1)C2 N1(C(c2c(CC)ncs2)=O)CCOCC12CCN(C(=O)C(C)=COC)C2 N1(C(c2ccn(C)c2)=O)CC(O)CC1C(=O)NOCCOCCN(C)C C1(CSCc2c(-n3cnnc3)ccc(F)c2)CSc2ccccc2O1 c1(NC(C)=O)ccc(C(=O)N(C)CCN)c(F)c1.n1(C(=O)NC2(CO)CC2)cccn1 Cc1cc(CN(C(=O)NCCc2ccc(O)cc2)CC2CCCO2)ncn1 Cc1cc(F)ccc1C(O)C(=O)NCC1(N2CCN(C)CC2)CCCCC1 N1(C(c2nc(C(C)OC)sc2)C(=O)N)CCC(OC)C12CCC2.C(C(C)C)C(=O)OC C(=O)(C(C1=CCSC1(C)C)N(C)C(C1CC1)C1CC1)NCCC(=O)OCC C(=O)(C(C)(C)CC1CC1)NC(CC)(C)CNC(=O)C=C(C)c1ccco1 c1(NCC)cncc(C(N2CCCCC2C(C)NC(=O)CC2CCCCC2)=O)c1 CC1CCN(C(c2[nH]ccc2C2CC2)=O)C(C)C1N(C(=O)CC1C=CCC1)CCO c1(C(N(CCCN(C(C(C)SCC(C)C)=O)C)C)=O)ccccc1OC(F)(F)F CCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)NOCCCO N1(C(C(COC)C)=O)CCC2OCCN(C(c3ccn4c(C)cnc4c3)=O)C2C1 O=C1COc2ncc(C(=O)NC3CCN(C(=O)CC4C=CCC4)CC3F)cc2N1 C1(CC(=O)NC(CNC(c2nc(C)n(C)n2)=O)(C)C2CC2)CCC(=O)NC1=O C1(C(=O)NC(C2CCCN2C(=O)C=Cc2cnc[nH]2)C)CCC(C(F)F)CC1 C(=O)(C(C)C1=CCCC1)N(C1CCN(C(c2ccccc2Cl)=O)CC1)CCOC c1(NC2CCN(C(Cc3cccc(C)c3)=O)CC2C)nc(C)nc2sccc12 C(=O)(CN=S(C)(C)=O)N1CCCC(C(C)NC(c2ccncc2F)=O)C1 C1(C(=O)NCCCCN(C)C(c2cc(N)cnc2Cl)=O)CCCC12CCC2 N1(C(C(C)NC(C)=O)=O)CCC2CN(C(C3CCCCS3(=O)=O)=O)CC2CC1 C1(O)(C(C)NC(c2ccc(CO)o2)=O)CCN(C(c2coc(C(F)F)n2)=O)C1 c1(C(=O)NC(CNC(C(CC)(C)CO)=O)(C)C)cncc2c1CCNC2=O c1(-c2cnc(CCC(=O)NCCCF)o2)cccc(-c2nn[nH]n2)c1 c1(CCC(=O)N(CC(CC)NC(c2n[nH]cc2F)=O)C)cc(F)c(F)c(F)c1 N1(C(C2(COC)CC2(F)F)=O)CCC(O)(C(C)NC(c2cnc[nH]2)=O)CC1 N1(C(CCC=CC)=O)CCC2(CCC2NC(c2ccc(OC)nc2)=O)CC1 C(=O)(CC1=CCN(C(=O)CCCCCC#N)CC1)OC.C12N(CC1(C)C)C2=O C1(NC(CCCC=C)=O)CN(C(=O)C(O)C(C)C)CC1(C)C N1(C(CC)=O)Cc2ccc(NC(=O)CC3CCC4(CCC4)O3)cc2C1 C(C(F)C(=O)NC1(C)CN(CCOC)C1)C1CN(C(C=CC=CCC)=O)C1 Cn1ncc([N+](=O)[O-])c1C(=O)NCCC(C)(C)NC(c1n[nH]cc1Br)=O c1(C(NNC(COCC2C(C)C2)=O)=O)c(O)nc(=O)n(Cc2cccs2)c1N CC1(C)C(C(=O)NCCOC2CCN(C(c3cc(C4CC4)ncn3)=O)C2)C1C#N c1(CC(N2C(C)CC(NC(=O)Cn3cc(Cl)cn3)C2)=O)ccc2c(c1)CC2 C12(NC(C3(C)CCCN3C(C3CCCC3)=O)=O)CCCN(CCC1)C2 CN1CC(c2nnnn2-c2ccccc2)(NC(C)(C)CCCN(C)C)CCC1=O C=O.CS(=O)CSCCCON.C1CC(CC)O1 c1(C(=O)NC(C2CN(C(=O)C(F)F)C2)C)cccc2c3c([nH]c12)CCC3 c1(CC(N2CC(NC(c3cncc(F)c3)=O)C2)=O)ccc(F)c(Cl)c1F C1(CNC(CCC(=O)NCCC)=O)CC2(CC2)CN1C(c1coc(Cl)n1)=O c1(OC)nc(=NC2CC(NC(c3c(Cl)ccc4c3OCO4)=O)C2)nc(OC)[nH]1 CC1(C)CN(C(C2(C)CCOC2)=O)CC(CNC(=O)CSc2cccs2)O1 C(=O)(C1CCCn2nccc21)NCC1(CNC(=O)Cc2n[nH]cc2Br)CCC1 c1(C(N2C(CNC(C3CCN(C(CC)=O)C3)=O)CC2)=O)cc(Cl)nnc1O N1(C(CNC(c2cc(OC)n(C)n2)=O)=O)C2CCCC1CN(C(=O)C=CCF)C2 c1(C(=O)NCCC2N(C(C(CC)C)=O)CCOC2)cnc2cc(Br)ccn12 N1(C(C(=O)NCc2cc(Cl)sc2Cl)=O)CCc2c(C(F)(F)F)n[nH]c2C1 C1(CNC(C(CC)OCC)=O)CC2CCC1N(C(=O)Cn1cnnc1O)C2 c1(C(=O)NCC2CN(C(c3c(SC)ccs3)=O)C(C)C2)c(Cl)ccc(F)c1N C(C1CCCN1C)=CC(=O)N(C1CN(C(=O)Cc2n[nH]cc2Br)C1)C c1(-c2c(F)ccc(OC)c2)ccc2c(c1C(=O)NCc1ccnn1C)OCO2 C1(NC(C2CC3(C2)CC(O)C3)=O)CC2C1CCN2C(c1ccc(Br)cn1)=O CN1CCC(N=c2[nH]ccc(=NCCN(C)C3CC3)[nH]2)c2ccccc21 N1(C(C(Cc2cccc(OC)c2)O)=O)C2CCC1CN(C(=O)C(Cl)=CCl)C2 C(=O)(CN=S(C)(C)=O)NCC1C(NC(C(c2nc(C)sc2)=O)=O)CC1 Cc1cc(C(=O)NCC(C2CCC2)NC(C2(C)C=CCC2)=O)nn1C(C)C1CC1 c1(CCC(=O)NCCOC2CCN(C(C3CCC3)=O)C2)cnc2ccccc2c1 C1(C(N2C(CC#C)CCCC2)=O)CC(O)CCN1C(=O)C(CSC)OC C(CC(C)CCNC(=O)CSC(C)(C)C)NC(c1cc(C)sc1)=O C1(OC)CCN(C(C2CCC(CNC(c3sccc3C)=O)CC2)=O)CC1C n1(CCC(=O)OC)c(NC=O)nnc1S(=O)(=O)c1ccc(NCCO)cc1 C(=O)(CCCCC(N)=O)N1CC(C)C(CNC(=O)CC2(O)CCCCC2)CC1 CC(=Cn1ccnn1)C(=O)N1CC(C)C(C)(CNC(=O)CNc2ncccn2)C1 CCC(CC)C(F)C(=O)NC1C2CN(C(=O)C(O)CC(C)(C)C)CC12 C1(C(=O)OC)CN(C(=O)CSCc2ncc(C(C)C)cc2C)CC1(C)C CC1=C(CNC(=NCc2cnsc2)NCC2CCOC2C)SCCO1 C(=O)(C(C)(C)C(C)(C)C)NC(C1CCN(C(CNC(CCC)=O)=O)CC1)CO C(=O)(C1CCCc2c(O)cccc21)NC1CCN(Cc2n(CCC)ncn2)CC1 c1(OCC(=O)NC(C2CC(C)C2)C)cccnc1 N1(C(C2(CCC)CCC2)=O)CC2(C1)SCCC2NC(c1oncc1C)=O c1(C(N2CCC(OC3CN(C(C=CC(N)=O)=O)C3)CC2)=O)ccn2ccnc2n1 CC1CCCC1(C)C(=O)NC1CCN(C(C2CC(=O)CO2)=O)CC1 C1(NC(c2c(OC)scc2)=O)CCN(C(=O)CC2CCC(O)C2)C1(C)C CC(CCCc1cccnc1)NC(c1cnnn1C1CCC1)c1nnnn1C N1(C(C(C)CF)=O)CCN(C)CC1CNC(c1csc(-c2cnn(C)c2)n1)=O C1(CNC(c2ccc(N(C)C)nc2)=O)CN(C(=O)CCc2cccs2)CC12CC2 N1(C(c2c(SC)n(C)nc2)=O)CCC(O)C(NC(=O)Cn2c(C)csc2=O)C1 C12(C(=O)NCCC3(NC(c4ccc(SC)o4)=O)CC3)CCC(C)(C1)OC2 C1(C(=O)NCC2(OC)CN(C(C3(C)CCC(F)(F)C3)=O)C2)CC2CC2CC1C CC1CC(NC(=O)C=CCCc2ccccc2)CCN1C(c1ccccc1)=O C(C(CC(C)C)C(=O)NC1(C)CCCN(C(c2ccnn2C(C)C)=O)C1)OC C(=O)(CCCCCC(C)C)NCC1N(C(CCCSC)=O)CC(C)(C)C1 Cc1nc(Cl)[nH]c(=NC2CC(C)N(C(c3[nH]cc4c3CCCC4)=O)C2)c1Cl c1(SCC)ccccc1CC(=O)NC1CN(C(C2C(C#N)C2(C)C)=O)C1 N1(Cc2cc(C)cc(C)c2O)CC2CCC1CN(C(C1CNC(=O)C1)=O)C2 c1(CNC(c2cnc(COC)s2)c2nnnn2CC2CCCO2)ccc(CO)cc1 N1(C(CN(C(=O)CC2CCCC2O)C2CC2)=O)CC2(CC(F)C2)C1 N1(C(COCC=C)=O)CCC2C(C1)CN2C(=O)C=CC1CCOCC1 c1(CC)ccc(C(N2CCCCC(N(C(=O)Cn3cc(C)cn3)C)C2)=O)c(C)c1 N1(C(CCSCC)=O)CC2(CCCCN2C(c2oc(CC)cc2C)=O)C1 C(=O)(C#CC1CCCC1)NC1CC(CNC(C(C)(C)SC)=O)C1(C)C C(C(C)(C)C(=O)N1CCN(C(=O)CNC(C2CCOC2)=O)CC1)OC(C)C C1(NC(C(C)OC)=O)Cc2ccccc2N(C(c2cnn(C(F)F)c2)=O)C1 C1(N(C(c2c(CC)non2)=O)C)CN(C(=O)C=CCN2CCCC2)CC1O CC(C(=O)NCC(c1ccccc1)N(C(=O)Cc1cccs1)C)S(N)(=O)=O C(=O)(C(C)CS(C)=O)N(CCCNC(c1c(C)nc(CO)o1)=O)C(C)C N1(C(Cc2cc(C)nn2C)=O)CC(C(N2CC3CC2(C(F)F)C3)=O)CC12CCC2 C1(CC#C)(NC(=O)C(c2cnn(C(C)(C)C)c2)C)CCN(C(C)=O)CC1 C1(C(=O)OC)(NC(c2c(O)cc(Br)cc2F)=O)Cc2ccccc2C1 CC1(C)OCCOC1C(=O)NCC1CC(NC(C2(c3ccno3)CCC2)=O)C1 c1(SC)ccc([N+](=O)[O-])c(C(=O)NCC(CC(C)C)NC(=O)C2=CCOC2)c1 CON(CC1CC1)C(=O)CC(C(F)(F)F)NC(c1cncn1C(C)C)=O N1(C(C2(N(C(C(C)=C(CC)C)=O)C3CC3)CCOCC2)=O)CC2(CCC2)OCC1C Cc1cc(=O)c(C(=O)NCC2CCCN2C(c2ccc(F)c(F)c2)=O)c[nH]1 c1(C(=O)NC2CC2CNC(C2CCCS2)=O)ccc2c(Br)cnn2c1 CCC(O)C(C)C(=O)NC1CCC(CN(C(=O)Cc2cncc(C)c2)C)CC1 C1(CNC(C=CC(CC)=CC)=O)CN(C(c2ncc[nH]2)=O)CCCO1 C(=O)(C(C)(C)CS(N)(=O)=O)N(CCN(C(c1cc(C(=O)OC)sn1)=O)C)C.C1CC1 CC(C)C(O)CC(=O)NCC1CC(O)CN1C(c1ccc(CO)cn1)=O N1(C(=O)CN2CCCCCC2)CCSCC1C1CC1 C1(C(C)C)CN(C(=O)C=Cc2ccsc2)CCN1C(c1ncccc1Br)=O c1(C(=O)NCC2COCCN2C(C2CC2C2CC2)=O)n[nH]cc1[N+](=O)[O-] C1(COC)CCN(C(=O)C(C)(N)C(F)F)CC12CCC2 CC1OC(C)CC1C(=O)Nc1cccc(NC(C2CCS(=O)(=O)N2)=O)c1 c1(C(N2CC(CC)N(C(=O)Cn3ccnc3C)CC2)=O)ccc2c(c1)NC(=O)C2 C#CC1(C(=O)NC(C)(C)CF)CCN(C(c2[nH]cc(C)c2C)=O)CC1 c1(C(N(C2(C(=O)NCC3(CC(C)C)CC3)CC2)C)=O)cc2cc[nH]c2cn1 C1(C(=O)NCCC(C)(C)NC(CC)=O)C2CCCC2CN1C(=O)OC(C)(C)C c1(C(N(CCNC(COc2ccn(C)n2)=O)C2CC2)=O)ccnc2ncccc12 C1(C(C(=O)NC(C)Cc2cnc[nH]2)C)CCN(C(c2cnc(Cl)n2C)=O)CC1 C(=O)(C1=C(C#N)CCC1)N1C(C(C)C)CN(C(C2C(C)CC(C)NC2=O)=O)CC1 C1(O)(CN(C(=O)CC(F)F)C)CCN(C(C2(CC3CC3)CC2)=O)CC1 c1(C(N2CCCC(C(=O)Nc3ccc(CC#N)cc3)C2)=O)ccc2c(c1)CNC2 Cc1nc(C(N2CCCC(N(C(C3(C)CCOCC3)=O)CC3CC3)C2)=O)[nH]c1C CC1CN(C(=O)CSC2CC2)C(C)CN1C(=O)COCc1csc(=N)[nH]1 N1(C(C2N(C(C(c3ccccc3)C)=O)CC(O)C2)=O)CCC(CC)C(O)C1 C(=O)(CCN=C(NCCN(C)C)N1CC2CC1CS2(=O)=S)Nc1ccc(C)cc1 C1(NC(C(C)C(F)F)=O)CCCCN(C(c2cc(Br)ccc2Cl)=O)C1 Cc1ccc(C(=O)NC2CC(F)(CNC(=O)CS(N)(=O)=O)C2)c(C2CC2)n1 C(=O)(C(C(C)(C)C)c1cc[nH]n1)N1CC(O)(CNC(Cc2c(C)nn(C)c2)=O)C1 c1(C(N2C3(c4cn(CC5(C)CCCO5)nn4)CC(C2)C3)=O)cc2c(cc1O)OCO2 c1(C(N2C3(CN(C(CCOCCN(C)C)=O)C3)CC2)=O)cc(C)cc(C)c1N Cc1cnc(CN(C(=O)C(CCOCCO)NC(=O)CC2CCCOC2)C)cn1 c1(C(=O)NC2C(SC)CN(C(C3(CCF)CCC3)=O)C2)ccc(C#N)c(C)n1 CCC(C)C(O)CC(=O)N1CCCCC1C(=O)Nc1ccc(C)cc1C c1(CC)ccsc1C(=O)NC(CNC(=O)C(CO)OC)CO Cc1c(CC(N2CC(NS(C)(=O)=O)C(F)C2)=O)cnn1CC(F)F N1(C(C(CCC)F)=O)CCN(C(=O)C(N2CCCCC2=O)C)C(C(C)C)C1 C1(=O)C(CC(C)C)N(C)C(=O)C2CN1CC2N(C)C.c1(CC)cn[nH]c1 N1(C(c2cc(COC)sc2)=O)CCC(NC(=O)CCn2cncn2)CC1C c1(C(=O)NC(CN(C(C(CC)OC)=O)CC)C)ccc2c(c1)CCCS2 CCCC(CC)NC(c1nnnn1C(C)(C)C)CCc1ccccc1 c1(COC(c2ccn(CCOC)n2)=O)cc(C)n(-c2cccnc2)c1C c1(C(N2CC3CCC(C2)N3C(c2cc(Cl)no2)=O)=O)ccc2c(c1F)CCC2 c1(-c2cc(NC(=O)NCc3cc(C(F)(F)F)cc(Cl)n3)no2)ccc(F)c(F)c1 c1(OC)ccccc1C(O)C(=O)NC1(CNC(=O)COc2ccc(Cl)nc2)CC1 C1(C(N(CCCC)CCCO)=O)(CNC(=O)CCn2cncn2)CCCCC1 c1(C(C)C(=O)NC(C)(C)CCNC(=O)C(C2CC2)C2CC2)ccc(F)cc1F CC1CC(C(=O)NC2CCCC2N(C2CCC2)C)N1C(c1nc[nH]n1)=O C(CN=c1nc(N(C(C)CC#N)C)cc(C)[nH]1)c1ccc(SC)cc1 c12cc(ccc1[N+](=O)[O-])S2.C(C(CO)NC(C1CCC1)=O)NC(C=CC(C)C)=O C(CC(C(C)(C)C)NC(=O)CC1(O)CCC1)N(C(CC1CCN(C)C1=O)=O)C C(N=c1cc(NC(=O)C(=O)NCCCS(C)=O)nc[nH]1)C1C(C)C1 N1(C(CCOC)=O)CC2CN(C(C3CCCN(C(C)C)C3)=O)CCC12 c1(C(=O)OC2CC(COC(CSC)=O)C2)ccccc1Oc1ccccc1 c1(C(N2CC(C(C(=O)NC(C)Cn3cncn3)OC)C2)=O)cc2n(n1)CCO2 c1(C(=O)NCCN(C(=O)CCc2cccc(Cl)c2)CCC)cc2sc(C)cc2s1 c1(C(N(CC(C)C(F)(F)F)C)=O)coc2c1CN(C(=O)C(=O)NCC1CC1)C2 c1(C(NNC(=O)Nc2cc(C(O)C(F)(F)F)ccn2)=O)ccc(Cl)cc1F c1(C(=O)NC2C(CC)N(C(C3CC(=O)NC(=O)C3)=O)CC2)cncc(F)c1C C(=O)(CC(C)(C)CC(F)F)N1CCC(O)(C(C)CNC(c2cc(N(C)C)no2)=O)C1 c1(CC(=O)NC(C2CCOC2)CNC(c2c(C)scn2)=O)cccc2ccsc12 c1(OCC)c(C)cnc(C(c2nccnc2C)NC(c2nnnn2C)C)c1C C1(CCCNC(CN)=O)CN(C(=O)CCOCCCN(C)C)CCO1.CC=O c1(OC(CC)C)cc(N2CCC(CO)(NC(=O)C(C)S(C)(=O)=O)CC2)nc(C)n1 C(=O)(C1=C(Cl)CCCC1)N1C(CNC(c2ccc(CC(C)C)s2)=O)CCCCC1 c1(CC(C(=O)OC)CNC2(C(C)C)CCC2)ccc(OC)c(O)c1 c1(NC(C2C(NC(c3c(F)cc(C)cc3F)=O)C2)=O)cncc(Cl)c1[N+](=O)[O-] N1(C(c2c(C)nncc2)=O)CC2(C1)CN(C(C1CC3(C1)CC(O)C3)=O)CCO2 Cc1cc(F)c(Cl)cc1C(=O)NCC1CCN1C(=O)CC1CCC(C2CC2)O1 C(=O)(C(CC(F)F)NC(=O)C(F)CC1CCOC1)N1CCC(CSC)CC1 N1(C(CSC(C)(C)C)=O)CC2(C1)CN(C(=O)Cc1ccn(C(F)F)n1)CC2CO c1(C(N2CC3C(CNC(C4CC4c4ncccn4)=O)C3C2)=O)cc(Cl)ccc1F c1(CN=C(NC(C=C)C)NC(C)C(C)COC)ccc(F)cc1F c1(CN(CC)CC)nccc(Cl)c1Cl.C1CCC(C)N1 N1(C(=O)NC2CC(C)N(Cc3ccccc3)CC2)CC2CS(=O)(=O)CC2(C#N)C1 CN1CCCC(NC(N2CCCC2Cc2ccc(Cl)cc2)=O)C1 c1(C(C(=O)Nc2cccc(NC(CC(C)F)=O)c2)(C)C)cccc2ccccc12 C1(N(C(C(C)OCC)=O)CC2CC2)CCN(C(C2(n3cncn3)CC2)=O)CC1 c1(OCC=C)cc(OC)ccc1C(=O)NC(C)CN(C(=O)CC#N)C C1(NC(C)C(=O)N2CC(CC(C)NC(C3CCOCC3)=O)C2)CCOCC1 CCC(C)C(C)N=c1[nH]c(N(C)CCc2cc(F)ccc2F)nc2c1CSC2 c1(NC(CSCCNC(C(C=C)(F)F)=O)=O)cccc(Cl)c1O C1(CC)C(C(N2CC(=O)CC2C(=O)N(CC(F)(F)Cl)C)=O)CCN1C Cc1cn2c(n1)CCC(N=c1nc3sccc3c(NCC(C)(F)F)[nH]1)C2 C1(CC(=O)NC2CC(n3cc(CCN(OC)C)nn3)C2)CCC(C)(C)O1 C1(CCNC(=O)C=CCO)CCCN(C(=O)CCc2ccccc2Cl)C1 N1(C(C(C)S(N)(=O)=O)=O)CCCC(O)(Cn2cc(Cn3ccnc3)nn2)CC1 C1(OC)CCCC(C(=O)NC2(CNC(c3cc(C)[nH]c3C)=O)CCCC2)C1 CCC(C)C(O)C(C)C(=O)NC1CC2(C1)CN(C(c1n[nH]cc1C)=O)C2 C(CC(=O)NCCCc1nnnn1C)(C(F)F)NC(c1n[nH]c(C)c1Cl)=O C(=O)(C(C)(C)NC(=O)CCc1nc(C(C)(C)C)no1)OCCC C1(C(=O)NCC(CNC(C2(CF)CCOCC2)=O)OCC)CCCCNC1=O Cc1onc(O)c1C(N1CC2C(CNC(C3CC(F)(CO)C3)=O)C2C1)=O N1(C(C(COC)N(C)C)=O)CCC(NC(=O)C(C)(C2CC2)NC(C)=O)C(C)(C)C1 c1(C(=O)NCC2(F)CC(CNC(C)=O)C2)ccc(C(F)(F)C(F)(F)F)cc1 c1(NC(C)Cc2ccn[nH]2)cc2c(s1)C(C)(C)CC2 C1(C(N(c2cnnc(O)c2Br)CCOC)=O)CC2(CC(C)=NO2)C1 C12CCCN1C2=O.CC(C)(O)CNC(=O)COC1CC(CCO)C1 C1(CCOC)CN(C(c2ccc(Cl)cc2N)=O)CCN1C(=O)C1=CC(C)(CC)C1 c1(CNC(c2ccc(OC)nn2)=O)ccc(CNC(C2CCCN2C)=O)cc1F CC(C)(CC(F)(F)F)C(=O)NC1CN(C(=O)C=CCO)CCC1O c1(NC(CC)(C)CO)ncc(C)cc1S(=O)(=O)NCC1CCCC12CC2 C1(C(=O)NCC(c2ncn(C)c2)O)CC(F)CCN1C(=O)CC1CC(C)(C)CO1 c1(C(C(N2CCC(CC(=O)Nc3n(C)ccn3)C2)=O)(F)F)ccccc1C#N C1(NC(=O)COC2CC(NC(c3c[nH]nc3-c3cccs3)=O)C2)C2CCCC12 C(c1cncnc1O)=CC(N1CCC(NC(c2c(Cl)cnn2C2CCCC2)=O)C1)=O C1(NC(C(CC=CCC)C)=O)CC12CCN(C(c1cc(C)cc(Cl)c1)=O)C2 c1(OC)cc(CCC(N2C3CCC2C(NC(=O)C=CS(C)=O)C3)=O)ccc1O C(CCCCN(C(=O)CCSCC(C)C)C1CC1)NC(C(C)=C(CC)C)=O C1(CNC(C2(C)CCCCC2)=O)CC2COCC2N1C(C1(C(F)F)CC1)=O CC1CC(C(=O)NC2C=CCN(C(c3sc(C#N)cc3Cl)=O)C2)CC(=O)N1 C1(CNC(c2c(C)cccn2)=O)CC2CCC(C1)N2C(C1CCCCN1C)=O C=CCCC(C(=O)NCCCN(C(=O)CC(O)C(C)C)C)NC(=O)OC(C)(C)C CC(C)(CNC(C1CC2CC1CC2=O)=O)CC(=O)NCC(O)C1(Cl)CC1 c1(C(N(C(CNC(C2C(C=C)OCC2)=O)C)CC)=O)cc(C)nc2[nH]nc(O)c12 c1(C(N(C2CCN(C(=O)C(O)CCC(C)C)C2)CC)=O)cc2cccnc2cn1 c1(CC)ccc(C)cc1NC(c1cccc(F)c1)c1nnnn1C1CCC1 C(=O)(CC(CNC(=O)C(C1CCCC1)OC)C1CCC1)NC(C#C)CCC c1(N(CCOC)C)cc(NCCN(C)CCF)nc(COC)n1 c1(CC(=O)NCc2cnc(Br)s2)cccc2nonc12 C1(C2CC2)(NC(C(CNC(C(CC)NC(N)=O)=O)N(C)C)=O)CCOC1 C1(CNC(CC2CC(=O)C2)=O)(CNC(C2CCC(CCO)CC2)=O)CC12CCC2 C1(F)(C(=O)NC2C(CC)CCC2)CCN(C(c2cncc(CO)c2)=O)C1 c1(C(=O)NCC2N(C(C3C(=C)C3)=O)CCC2C)c(CC)ncnc1CC C(=O)(C1=NOC2(CCOC2)C1)N1CC(CCNC(C2(SC)CCC2)=O)OCC1 C1(CCOC)CN(C(C2(n3ccnn3)CC2)=O)CCN1C(c1cccc(F)c1)=O N1(C(C)C)CCOC(C(=O)NCC(C2CCCCN2C(=O)CNC(N)=O)(C)C)C1 C1(C(=O)NCCN2CC3CC3C2)CCOCCN1C(=O)CCC(F)(F)F N1(c2cccc(C(N)=O)n2)CCC(N=C2C=Cn3ccnc32)C1 C=Cc1ccc(C(=O)NCC2CC2NC(c2ccc(Br)nc2OC)=O)cc1 C1(NC(c2cccc(C3CC3)c2)=O)CCCCCC1NC(=O)C(O)CC1CC1 Cc1ccc(NC(c2sccc2CNC(C2(C)CNC(=O)C2)=O)=O)c(C)n1 c1(OC)ccc2c(c1)OCC(C(N1CCC(C)(NC(=O)CCOC3CC3)C1)=O)C2 C1(C(=O)NC(C2N(C(c3c(CC)n(C)nn3)=O)CCC2)C)CCC=CCCC1 c1(C(=O)NCC(CNC(C(C)(C)C)=O)F)c[nH]c2nc(Br)ccc12 C1(CC)(CNC(C2(C)CCN(C(c3cnn(C(F)F)c3)=O)C2)=O)CCC(=O)N1 C1(CCNC(C2CC2(F)F)=O)CCCN1C(=O)CC1CCSC1 N1(CCC(=O)NCCCOCCNC(C(CC)F)=O)CCCC(N(C)C)C1 CCC(C)(CO)C(=O)NC1CCN(C(c2ccnc(OC(C)(C)C)c2)=O)C1 C1(CNC(C(C)(C)n2ccnn2)=O)CN(C(=O)CC2CCC(=O)NC2)CC(C)(C)O1 N#Cc1ccc(S(=O)(=O)N2CCCOC2)cc1NC1CCC1c1ccccn1 C1(NC(CC2(NC(C)=O)CC2)=O)CN(C(=O)C(C2CCCCC2)C)CC1C c1(OC)c(C(N2CCCCC2CNC(=O)CN(C)C(N)=O)=O)cccc1[N+](=O)[O-] CN1CCN(C(=O)C#CC2CCC2)CC1c1cn(CC2CC2C(F)(F)F)nn1 C1(C(=O)NC(C(CC)C)C)CC12CCN(Cc1cccc([N+](=O)[O-])c1)CC2 C1C(F)(F)CCC(=O)NCC2(CCCCC2)c2cn1nn2.CC(F)CC(=O)N(C)C C1(O)(CC(C)NC(=O)CC2(c3ccccc3)CCCC2)CCN(c2nnco2)C1 C(=O)(C1CSc2ccccc21)N1CC(C2(NC(c3cc(C)oc3)=O)CC2)C1 C(CC(O)C(=O)N1CCC(NC(=O)C2CC2)CC1)NC(CC1(C=C)CCC1)=O c1(CCN(CC)CC)cc(-c2nnc(CN(C)C)o2)sc1C c1(C(=O)NC(C2CCOC2)CNC(c2cnc(SC)[nH]2)=O)cccc(F)c1 Cc1cc(C(N(C)CCNC(=O)C(C)C(C)C)=O)cnc1O C12(CNC(c3nnnn3CC3CCCCC3)(C3CCCC3)C)CCC(CC1)C2 N1(C(c2ccc(Cl)cc2)=O)CCCN(C(C2CC2Oc2ccccc2)=O)CC1 N1(C(CC2C(C(=O)OC)C2)=O)CC2CN(C(C3(O)CC4CCC3C4)=O)CC2(C)C1 N1(C(CC(CC)C(C)C)=O)CC(CO)C2(C1)CN(c1ncnc3n[nH]c(C)c13)C2 C1(C(=O)NC(C)CCCNC(=O)C=Cc2ncco2)OCCOC1C C12(C(NOCCC(C=C)C)=O)C(NC(c3nccnc3OC)=O)C3CC1C2C3 Cc1c(C(=O)NCC2(C(F)F)CCN(C(=O)C(F)=C3CCCC3)C2)cccc1O C(=O)(C(F)C(F)(F)F)NCCOCCC(=O)NCC(C)(O)C1CCC1 c1(N2C(CCNC(c3ccc(COC)[nH]3)=O)CCCC2)nc(C)nc2[nH]ccc12 N1(C(=O)OC(C)(C)C)C2CC1CN(C(=O)C(C1CC3CCC1O3)=O)C2 CC1(CNC(c2ccccn2)=O)CN(c2cc(C(N)=O)ncn2)CCO1 c1(C(N2CC(NC(COCC(C)C)=O)C(CC(C)(C)C)C2)=O)ccc(O)nc1Cl Cc1[nH]nc2ccc(C(N3CC(O)(CNC(C4(C(F)F)CCC4)=O)C3)=O)c(Cl)c12 c1(C(=O)OCC)cccnc1NC1CCN(C(=O)C2=CCCS2)CC1 C1(O)(CNC(C(C)=CC)=O)CCCN(C(=O)C(C(C)C)NC(=O)OC(C)C)C1 c1(C(=O)NC2C(NC(C=C(C)C)=O)CCC2)sc2nccn2c1C C#CC1CCCCN1C(C1(OC)CCN(C(=O)CCc2cncs2)C1)=O C1(OC)CCN(C(C2(CF)C=CCN2C(c2cc(CC3CC3)on2)=O)=O)CC1F N1(C(CCSCC(C)C)=O)CCC(CNC(C2(Cl)CC2)=O)C(O)C1 CC1CCC(NC(=O)CC2CC(C)(C)C2)CN1C(=O)CCOCCOCCO CC1(C)CN(C(=O)CCn2cnnn2)CCC1C(N1CC(CO)C2(CC2)C1)=O Cc1ccc(C(N2CCC(N(C)C(C3CC(CCF)C3)=O)C2)=O)s1 C(=O)(CC(C)(C)C(F)F)NC(C1CCCCC1)C(N1CCCC(OC)C1C)=O N1(C(COc2ccc(C)cc2)=O)CCC(C)C(CNC(C2(O)CCC2)=O)C1 CC1CN(C(=O)Cc2cscn2)CC(C)C1NC(=O)C(N1CCN(C)CC1)C N1(C(c2c(C)ccnc2C)=O)CC2COCCC2(NC(c2nn[nH]c2Cl)=O)C1 c1(CC=C)c(C)c(C(=O)COC(C2CC3(CN2)CC3(F)F)=O)n2ccccc12 c1(CC)ccc(C(COCc2ccccc2)C(=O)NCCCCl)cc1 C1(NC(CC=CC)=O)CCCC12CCN(C(c1cc(CC)on1)=O)CC2 C1(c2nc(CC)nn2Cc2cccc(Cl)c2)CCc2nncn2CC1 c1(CN(CC)CC)ccccc1F.c1(C(=O)O)cn(CC(F)F)nc1C N1(C(Cc2ccc(S(C)=O)cc2)=O)CCC2(O)CCCCC2C1 C12CCN(CC1O)C(=O)CCCONC2=O.c1(C=O)ccc(F)cc1.CO c1(C(N2CCC(NC(C(C=CC)O)=O)C(F)C2)=O)cc(N=S(C)(C)=O)ccn1 C1(NC(c2c(C)cno2)=O)CC2CC(C1)N(C(c1ccn3ccccc13)=O)C2 c1(C(=O)NC(C(=O)OC)CF)ccc(N)c(Cl)c1 C1(N(C)C(c2coc(C(N)=O)c2)=O)CCC(NC(c2ccncn2)=O)CC1 N(C1CN(C(C2(CO)CCOCC2)=O)Cc2ccccc21)C(C=NOC)=O c1(C(=O)NCC2CCN(C(C(CC)C(C)(F)F)=O)C2)cc2n(n1)CCNS2(=O)=O C1(CNC(c2c(C)ccs2)=O)CC(C)(C)CN1C(=O)C=CS(C)=O C1(NC(=O)Cc2c(F)cccc2F)CC2CC1N(C(=O)CCc1ccon1)C2 c1(N2CC(C)C(C)(CO)C2)ncc(S(=O)(=O)NCc2ccns2)cc1Cl CCC(CC(=O)NC1CCCC1)N(C(=O)C(C1CCOCC1)C)CCOC C1(C(N(CC=C)CCOC)=O)(CNC(=O)C(c2ccn(C)c2)C)CCCCC1 C1(C(=O)NC(C(C)C)CNC(C2C=CCCC2)=O)COc2ccccc2O1 Cc1cc(Cl)ccc1C(=O)NCCC(C)N(C)C(C1CCN(C)C1C)=O CCCCCC(F)C(=O)N1CC=CC1(C(=O)NCCCCCCCO)COC C1(COC(c2c(C)nn(C(C)C)c2C)=O)CCN(C(=O)Cc2cccs2)C(=O)CO1 n1(CC(N2CC(N)(NCc3cccc(OC)c3)C2)=O)cc(C)ccc1=O N1(C(CC=C(C)C)=O)CCC(C)(C)C(C(=O)NC(C2CC(F)(F)C2)C)C1 C1(NC(C2(CNC(C=C(C)C3CC3)=O)CCC2)=O)CCC(CN(C)C)C1 CC1(C)CC(NC(=O)CC(F)F)CCN(C(C2CC3(CCOCC3)C2)=O)C1 C(CC(C)(C)C)(C(=O)N1CCCCC1CCC(=O)NCCOCC(F)F)OC c1(CN)cccc(COC(c2cccnc2OCC(F)F)=O)n1 C1(C(=O)NCC2(CN(C(C3(CCC)CCC3)=O)C)CC2)CC2(C1)CC(F)C2 CN1CCC(N(C(=O)CC=CCNC(c2ccnn2C)=O)C)CC1 N1(C(=O)CN2CCCCC2=O)CCNC2(CCNCC2)C1 N1(CC(=O)O)C(=O)CC(NCC(O)CC2CC2)C1c1cccnc1 c1(C(=O)N(CC(N2CCCC2)=O)C2CC2)sc2cc(Br)ccc2c1Cl c1(C(=O)OCC)ccc(NC(=O)C(=O)NC(C2CCN(C)C2)C)c(Br)n1 C(CCC(C)C(=O)NCC1CN(C(C2CC(=O)N2)=O)CC1C(F)(F)F)OC CCCCC(C(=O)NCC1CCC(=O)N1)NC(c1ncc(C)cc1F)=O N1(C(C2N(C(Cc3ccc(C)o3)=O)CC(C)CC2)=O)CCC2CC1C(=O)O2 N1(C(CC2C(C(=O)OCC)C2)=O)CCC(C)(CNC(=O)CCC#N)CC1 C(C(C)C(C)C(=O)NCC1(NC(C2CC3(C2)OCCO3)=O)CCCCC1)OC c1(C(N2C3CCC(NC(C(CC)(F)F)=O)C(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 CN1CC2(CCN(C(C3CCC4(CC3)CC4(F)F)=O)CC2CO)C1 c1(-c2cc(C(=O)NCC(C3CCOC3)NC(C=C(C)Cl)=O)no2)ccccc1F C=CCC(C(=O)NC1(CNC(c2cn(C)nc2C)=O)CCCCC1C)C(C)C c1(OC)cccc(CNC(=O)C(c2sccc2I)N2CC3CC3C2)c1 C(CC(C)C(=O)NC(Cc1ccoc1)C(=O)NCc1cnnn1C)=CCC N1(C(C(CC=C)(C)C)=O)CCC(C2CCN(c3nncs3)C2)CC1 Cc1nn(CC(=O)N(C)CCNC(=O)Cc2ncsc2Cl)c(=O)o1 CCCC(CCCNC(=O)CCCC1CCC1)NC(C1CC(OC)C1)=O C1(CNC(CCCc2onc(CC)n2)=O)CN(CCC2CCCO2)CCCO1 CC(C(=O)N(C1(C)CC1F)C1CC1)C1CCOC1 c1(C(=O)NCCCC#C)cc(CN(C(=O)C=CC2CCC2)C2CC2)ccn1 C(C(CC1CC1)C(=O)N1CCN(CC2CC2)CC1)NC(C1CC12CCC2)=O C1(CNC(C(C)(C)OC)=O)CC(NC(c2ccc(SC(F)(F)F)cn2)=O)C1(C)C N1(C(c2c(CC)cccc2)=O)CCC2(CCOC2)C(CNC(C2(C)CCC2)=O)C1 N1(C(c2c(C)scc2)=O)CCOC(CC(N2CCC(CN=[N+]=[N-])C2)=O)C1 C(C(F)(C(=O)N1CC2(CC2)CC1C)C(C)C)NC(CCc1cc(C)[nH]n1)=O C=CCC(CNC(=O)C(C1CCCCC1)C)C(=O)Nc1cnc(C)nc1 C(=O)(C(C)(C)CNC(C)=O)NCC1OCC(C(N(c2ccccn2)CC)=O)C1 N1(CC(O)CF)CCN(CCCC2(c3ccncn3)CC2)CC1 c1(C(COC)NC(C23CC(n4cc(C(C)NC)nn4)C2C3)=O)cccc(OC)c1 c1(C(=O)NCCCN(C(c2cnn(C(CC)C)c2C)=O)C)nccc(C#N)n1 C1(CCC2N(C(CCOCC#C)=O)CCC2)CCCCN1C(C1(Cl)CC1(F)F)=O C1(C(=O)OC)C(C)CCCN1C(C1CC2(CCC2)CO1)C(=O)NCCC#N C1(C(=O)NC(C2(OC)CCC2)C)N(C(=O)C2=C(C)CC2)CC12CCCC2 C(=O)(CCCC(=O)N1CC2CC1(C(=O)Nc1cc(C)cnc1O)C2)OCC c1(C(C)C)ncc(C(=O)N(C(C)CNC(=O)CC2CCC2(C)C)C)s1 N1(C(c2c(C)nn(CCO)c2C)=O)CCN(c2ccnc(CO)n2)C(C#N)C1 N1(C(C2C3CCCC23)C(=O)NCCSC)CCC2(CCCN(C)C2)CC1 C1(C(=O)NCC(C(=O)OCC)C)CC1C1CN(C(C2CCC3(CC3)C2)=O)C1 c1(C(N2CCCC(NC(Cc3cc(C(C)C)no3)=O)C2)=O)cc(N)c(Cl)c(O)c1 c1(C(N(CC(O)CNC(c2cocn2)=O)C)=O)nc(Br)c2ccccn12 C1(CC)(CC)CC(NC(C2C(Cl)(Cl)C23CC3)=O)CN1C(=O)CC1(CSC)CC1 c1(CN(CC(=O)NC2CCN(C(CC(C)N(C)C)=O)C2C)C)ccccc1Cl c1(C(C)NC(C2CCCC(C(=O)O)C2)=O)nc2cc3c(cc2[nH]1)OCCO3 C1(NC(CCC)=O)CN(C(=O)C=C(C)CN2CCOCC2)CC2(CCC2)C1 c1(C(N(C)CC2(CNC(C(C)n3cncn3)=O)CC2)=O)ccc(CO)s1 O=C(C1=CC2(CCN(C(C3CCSC3)=O)C2)C1)NCc1cc(CO)ccn1 CC1CN(C(C2CC3(CCC3)CN2C(=O)CC2=CCC2)=O)C(C)C(C)(C)O1 c1(C(N(C2CN(C(c3c(CC)nco3)=O)C2)C)=O)cccc(N2CCNC2=O)c1 C(C)(C(=O)C(F)(F)F)OC(C(CCc1ccccc1F)SC)=O C(CC(F)F)(C(=O)NCC(C)CC1CC1)N(C(c1nc(C)c(C)s1)=O)C C1(C#N)(CC(=O)NC(CN(C(C(C)OCC)=O)C)C)CCCCC1 C#CCCCCC(=O)NC1(C)CCN(C(c2ccc(C#C)nc2)=O)CC1 N1(C(ONC(c2c(C)non2)=O)=O)CCC2C(CCN2C)C1.c12nnn(C)c1C2 C1(C)(CNC(c2cc(C)cc(O)n2)=O)COCCN(C(=O)Cc2ccsc2C)C1 N1(c2ccc(C#N)cn2)CCC2(NC(c3conc3C3CC3)=O)CCCC12 C1(NC(CC(c2cccc(Br)c2)C)=O)CCC2CN(C(c3cccs3)=O)CC2C1 N1(C(C(C#N)c2ccccc2)=O)CCCC(NCc2nccnc2Cl)CC1 N1(C(=O)C=CC2CCOCC2)C(CC(=O)NCC(O)CC(F)(F)F)C2CCCC12 C1(CN(C)C(c2csnn2)=O)CCCCN1C(c1ncncc1Cl)=O c1(C(CCC)=O)ccc([N+](=O)[O-])cc1-c1ccc(NC(c2ccccc2)CC)s1 N1(C(C(F)=CC)=O)CCN(C(c2cc(C(N)=O)ccc2C)=O)C2CCCCC2C1 N1(C(c2c(C)c[nH]n2)=O)CC2CCC2(CNC(=O)Cc2cccc3nsnc23)C1 c1(C(N2C(C)CC(NC(CC3CC(OC)C3(C)C)=O)C2)=O)ccc2c(c1)CCN2 N1(C(CC=CCC)=O)Cc2n[nH]cc2C1C(=O)NOCCC1CC1 c1(C(=O)NCC(CC(C)C)NC(=O)C(C)CF)c(O)cc(F)cc1F C1(CNC(c2n(C)ncc2)=O)CN(C(c2ccccc2F)=O)CC1(F)F C1(CNC(CCCC#C)=O)CN(C(=O)CN2CCCCC2=O)CC12CCOCC2 C(=O)(N1CCCc2ccnn21)C1CC(CC)C1(C)C.c12occc1CNC2=O C1(NC(c2c(CC)ccs2)=O)CN(C(C2COC(=O)C2)=O)C2(CCC2)C1 C=C=C(C)CC(=O)NC(C)C(C(C)C)NC(c1cc(OC)n(C)n1)=O C1(C(=O)NCCCOCCCC)(NC(=O)C(CC)OCC)CC1(C)C C1(C(=O)OCC)CCC(CN2CC(F)CC2C(=O)NCCc2cnn(C)c2)CC1 S(=O)(=O)(c1ccc(Br)cc1NCC(O)C1(Cl)CC1)NC(C)CC1CCCO1 c1(NC2CCCN(C(C(CCC)NC(N)=O)=O)C2)nnc(C)cc1C(=O)N(C)C c1(C(=O)OCC2C=CCC2)cc2c(F)c(F)c(Br)cc2[nH]1 N1(C(c2cc(C(C)C)no2)=O)CCC(C(F)F)(CNC(C2C=CCCC2)=O)C1 n1(CCC(=O)NC2(C)CN(c3ccncn3)C2)ncc2c1CN(C(=O)CO)C2 C1(C(=O)NC23CC(CNC(C4CCS4(=O)=O)=O)(C2)C3)(OC)CCCC(C)(C)C1 CC(C)C(F)(CNC(=O)C1=CCCC1)C(=O)N1CCSCCC1C c1(C(=O)NCC2CCCN2C(=O)CCc2ccc(Cl)nc2)cccc2ncnn12 c1(CNC(c2ncc(COC)s2)c2nnnn2C2COC2)c(Cl)c(SC)nn1C Cn1cc(C(=O)NC2CCCN(C(=O)CC3CC4CCC3O4)C2)cc1Br N1(C(c2cn3c(n2)C(=O)N3C)=O)CCCC(C2(NC(C3CCC(=O)N3)=O)CC2)C1 C12(CNC(c3c(CCC)occ3)=O)CCCC1CCN2C(c1cccnn1)=O N1(C(CCC=C=C)=O)CC2(CCN(C(c3cnc(Cl)s3)=O)CC2)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCCOC(CCNC(c2ncoc2C2CC2)=O)C1 O=C(C#CC1CCCCO1)NCC(C1CCC1)NC(c1ccc2sccc2c1)=O C#CCC(C(=O)OC)NC(=O)CC1C(NC(C2CC2(Cl)Cl)=O)CC1O c1(C(=O)NCC(C)C(=O)NC2CC(O)C(O)C2)cnc(S)nc1 c1(OC)c(C(=O)NCC2(O)CCN(C(c3cnsn3)=O)C2)cnc2ccccc12 C1(CNC(C=CC)=O)CC2COCC2N1C(c1nccn1C)=O CC1CC(C(=O)N2CCC=C(CNC(C3CC(C(C)C)C3)=O)C2)=NO1 C(N=c1cc(C)[nH]c2ccc(N)cc12)C1C(c2c(C(=O)OC)c(F)ccc2)C1 N1(C(C(C)CC(F)(F)F)=O)CCC2(CC1)CCN(C(C1CC3CCC3C1)=O)C2 C(C1=CCN(C(=O)C2=CCCCO2)CC1)NC(=O)CC1CC2CCC1C2 c1(N2CCC(C)(NC(CCOCC#C)=O)C2)cc(C)nc2c(C)cnn12 c1(CNC(C2(NC(C=CC(=O)OCC)=O)CC2)=O)cccc(Cl)c1 c1(CN(C)C(C2CC(F)(F)C2)=O)nnn(C2CC2)n1 C(CCC)(C(=O)N1CCC(N(CCO)C(C2CC(F)C(=O)N2)=O)CC1)=CCC CC(C)(CONC(c1cc(O)ncc1F)=O)CC(=O)NC1CN2CCCC1C2 C12(NC(c3ccc(=O)n(CCO)c3)=O)CCOCC1CN(C(C1CCCC1)=O)C2 N1(C(C(CC2CN(C(CN(C3CC3)OC(C)=O)=O)C2)F)=O)CCOC(C(C)C)C1 c1(C(=O)NCC2N(c3nc(C)cc(C(=O)OC)n3)CC(F)C2)cc(Cl)c(F)cc1F C1(C(N(C2CCN(C(C3CCCOCC3)=O)C2)CCO)=O)CC2(C1)CC(F)(F)C2 c1(OC)c(C)cc(C(=O)NCC(O)CCNC(=O)C(C)n2cnnn2)cc1Cl C12(NC(CC(CC)CN(C)C)=O)CC3CCC(C1C2)N3C(=O)CC1CN(C)C1 CCCCCC(O)C(=O)N(C1CCN(C(c2cc(C#N)ccc2O)=O)C1)CC Nc1ccc(C(=O)NCC2CC(NC(c3ccon3)=O)C2)c([N+](=O)[O-])c1 C1(NC(CSc2nc(C)c(C(=O)OC3CC3)s2)=O)CCCCN(C(=O)C(C)CO)C1 N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)CC2CCCC2(F)F)CC1c1cn[nH]c1 N1(C(Cc2scc(C)c2)=O)CCCC(F)(C(=O)NCCNc2cccnc2)C1 O=C1CC(C(=O)N2CCN(C(C3(F)CC3)=O)CC2)c2ccccc21 N1(C(c2c(CC)csc2)=O)CC2COCC2(C(=O)NCc2ccc(C)c(O)n2)C1 C1(C(N(CCC(=O)NC2CCOCC2F)CC=C)=O)CCC(=O)N(C)C1 CCCCCC(C)(c1nnnn1-c1ccc(OC)cc1)NC(c1ccccn1)C C(=O)(CCCC(=O)NCCc1cccc(O)n1)NC CC1CN(C(c2cncnc2)=O)CCCN1C(=O)CC1CCCCCC1(F)F C1(C(=O)NC(CCNC(C)=O)(C)C)CCCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 c1(C(C)CC(=O)NC2CC(C)(NC(=O)CCN3CCCC3)C2)ccc(F)cc1 C(=O)(C1=COCCO1)N1CC(CNC(C2C(C(=O)OC(C)(C)C)CC2)=O)C(O)C1 c1(N(CC(NC2CCN(c3c(Cl)ccc(C)c3)C2)=N)C)nncc2ccccc12 Cc1nn(-c2ccnc(F)c2)cc1CN1CCCC(NC(=O)OC(C)(C)C)C1 c1(C(=O)NCC2C(NC(C(C)OCCCC)=O)COC2)nccc(Cl)c1Cl C(=O)(CCCC(=O)NCC(=O)NCCOC1(C)CCCC1)OCC N1(C(C2C(CCC)CCC2)=O)CC2CC(CNC(c3ccc(Cl)c(F)c3)=O)C2C1 C1(CNC(C(CC)N(C)C)=O)CN(C(c2cc(F)c(F)cc2Cl)=O)CC(C)(C)O1 c1(C(=O)NC2CC3CC2CN3C(c2cccc(=O)o2)=O)cc2c[nH]cnc-2n1 CCCC(CC(=O)NC1C=CC(C(=O)NCc2nc(CC)no2)C1)C(C)C Cc1cc(C(=O)NCC2CCN2C(=O)C2=NNC(C(F)(F)F)C2)ccc1Cl C1(COC)CN(C(c2ccncc2SC)=O)CCN1C(=O)C(CC1CC1)OC C(C)(CSC)(C(=O)N(C1(CC(C)C)CC1)C1CC1)NC(C(C)OCCC=C)=O c1(C(N2CC(C(Cn3cc(CCCSC)nn3)F)C2)=O)cccc2c1OC(C)C2 N1(C(C2CCSC2)=O)CCC2C(C(=O)NCCCc3nncs3)C2C1 c1(CC)ccc(CCC(=O)NCC(C(C)C)NC(=O)C(C)SC)cc1 CCC(F)(F)CC(=O)N(C)CCOCCNC(c1cc(OC)ncc1Br)=O N1(C(c2n(CC)c(O)nc2)=O)CC(CN(C(=O)Cn2nnnc2C)C)C2(CC2)C1 N#Cc1ccc(NC(C2CN(C(=O)Cc3ccc(Br)nc3)CCN2)=O)cn1 N1(C(C2(COC(C)C)CC2)=O)CCN(C(C2CCCS2)=O)CC(C)C1 C1(C(=O)NCC2CCN(C(C(C(C)C)N(C)C)=O)CC2C)CC2CCCCN2C1 Cc1ccc(CC(N2CC3CC2CN3Cc2ccc(O)c(C(C)C)c2)=O)c(C)c1 CCCCC(CCCC)C(=O)NC1CC(C)(NC(C2CC(F)C(=O)N2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)N.N12CCCC1C(C1CC1)C1(CC1)CNC(=O)C2.CO C(C(C)(C)CC(=O)NC1(c2nc[nH]n2)CC1)NC(CC(C)(F)F)=O c1(CC)cc(C(=O)NC2CC(c3ccncc3)C2)cc2c[nH]nc12 c12ccc(cc1)C(=O)N1CCCC1C(C)CCO2.c1(CC(=O)NC)ccno1 CC1=C(C(=O)N2CC(C3CN(C(c4ccc(C)s4)=O)C3)C2)COCC1 C(CC)(CC)(CCNC(=O)CCC1CCCC(C)(C)C1)NC(COCCC=C)=O c1(CC)cc(F)c(C(=O)NCCNC(=O)CCc2cnc3ncccn23)cc1F CCC(C)(CO)C(=O)NCC1CCN(C(c2c(C)nn(C(C)(C)C)c2Cl)=O)C1 c1(C(N(C2CN(C(CC(O)CO)=O)C2)C)=O)c[nH]nc1-n1cccn1 N1(C(COc2ccc(CC)cc2OC)=O)CC2CCC(C1)N2C(=O)C(O)C1CC1 CC(C)C(O)C(C)C(=O)NC12CC(CNC(c3cnc(O)cc3O)=O)(C1)C2 N1(C(C2(CC(C)C)CC2)=O)CCC(C)C(CNC(=O)CC2(C#N)CC2)C1 CCC(CC)CC(F)C(=O)NC1CC1NC(c1cccc(F)c1C)=O Cn1c(C(N2CCCC(CCNC(C3(n4cccn4)CCC3)=O)C2)=O)cnc1O C1(CC(=O)NC23CC(O)C2C3)CC2(CCC2)CO1 C=Cc1cncc(C(=O)N(CCNC(=O)C(C)CC(F)F)CCOCCO)c1 c1(N2CCN(C(C)C)CC2)nc(=NCCCCCCO)[nH]c2c(F)cc(F)cc12 C1(C)(C(=O)NC(CNC(c2c(CC)[nH]cc2)=O)C)CC(C#N)C1 C1(C(N2CC(NC(c3c(NC)scn3)=O)(COC)C2)=O)CCC(=O)N(C)C1 c1(C(N(c2c(C)cncn2)C2CC(N)C2)=O)c(C)c(C)nn1C c1(NC(=O)OC)ccc(-c2ccccc2N2CCC(O)C2)cc1 N1(C(COC(CC)C)=O)CCC(O)C(N(C(=O)C(C)Cn2ccc(C)n2)C)C1 c1(N(C(C)CNC(=O)CSc2ccncc2)C)ncc(Cl)c(C(=O)N(C)C)n1 CCCCCCCCN(C(=O)C(CC1CC1)NC(=O)C(C)=C(C)C)C CN1CCC(C(=O)NCC2(O)CC(CNC(=O)Cn3ccc(C4CC4)n3)C2)C1=O CCCC(C1CC1)NC(=O)C(C1CCCO1)NC(=O)CNC(=O)CN(C)C Cc1cc(C(N2C(C(=O)NC3(C4CC4)CC3)CCC2C(C)C)=O)cc(O)n1 c1(C(=O)Nc2cc(I)ccc2F)n[nH]c2c1CN(Cc1ccc(O)cc1)C2 N1(C(C(N)=O)=O)CCC2(CCCCN(C(C3CC4CC4C3)=O)C2)C1 C#CCCCCCC(=O)NC1CC2(C1)CC2NC(C12CC(C)(C1)C2)=O c1(NC(C(=O)NCC)(C)C)nc(C)cc(=NCC2CCCC(C(F)(F)F)C2)[nH]1 N1(C(=O)NCc2ncc(Cl)cn2)C(CO)CCC12CCC2 C1(N(C(c2c(C)coc2)=O)C)CN(C(=O)CCCc2csc(=N)[nH]2)CC1O c1(C(C)=O)ccc(CC(N2CC(O)(C3CCCN3C(=O)Cc3ccno3)C2)=O)s1 c1(N(CCC(N)=O)C)nc2c(c(=NCC3(C)CCCCC3(F)F)[nH]1)CC(C)CC2 C(C)(CO)(CC(C)C)NC(COC1CC(NC(c2cc(C)sc2)=O)C1)=O Cc1sc(C(N2CC(CNC(=O)CC3CCC3)C3(CC3)C2)=O)cc1[N+](=O)[O-] C1(=O)C(CCCC)O1.O1NC(=O)C2CCC2CC1.C#CCOC=C Cc1ccc(CN(C)C(c2c[nH]nc2CNC(c2ccccc2Cl)=O)=O)cc1 c1(C(N2CCC(NC(COCC)=O)C(C)C2)=O)cnc(O)c2cccnc12 c1(SCC23C(C(=O)OCC)OC(C)(C2)C3)cc(OC)c(OC)c(OC)c1 C(=O)(CCCCCCCO)N(c1nc(N(CCCF)C)nc2sccc12)C N1(C(C2CC(CC)C2)=O)CCC(NC(c2cc(CO)[nH]n2)=O)C1C(C)C c1(C(=O)NC2(CC=C)CN(C(=O)CCC(C)C)C2)cc(O)nc(N(C)C)n1 C1(C(N(C(CCCC)C)C)=O)CCCCN(C(=O)C(c2cncnc2)C)C1 C(C(=O)NCC1(n2cccn2)CC1)(C(C)(C)C)n1cc(C(CC)O)nn1 C(=O)(C(C)CC(=O)N1CCC(C)C(NC(=O)C=Cc2ccncc2C)C1)OC N1(C(CC)=O)CC2(NC(=O)CC(=O)NCC3CC3)CC1C2 C(=O)(C(C)(C)CC(C)C)NC(C1CCN(C(Cc2cc(C)c(CO)cc2)=O)C1)C C1(NC(c2cnc(COC)s2)=O)CN(C(C2CN(C)C(=O)N2)=O)CC2CC12 c1(N(c2ccc(C)cn2)C(c2cc(Cl)ncn2)=O)n[nH]c2c1CNC2 C1(NC(c2ccc(C(C)C)s2)=O)CCN(C(=O)C(C)CC(F)(F)F)CC12CCC2 N1(C(C(CC=C)NC(c2cnc(O)c(F)c2)=O)=O)CCC(C2=NOCC2)C1 C1(CN(C)C(c2cc(-c3ccns3)on2)=O)CCCN(C(C2CNC(=O)N2C)=O)C1 N1(CC(N2CCC(COC)(NC(=O)CSc3ccccn3)C2)=O)CCS(=O)(=O)CC1 C(CCCCCC(=O)N1CCCC12CCOC2)NC(C(CC)N(COC)CC)=O c1(C(=O)NC(C)CCCNC(c2ccoc2C(F)(F)F)=O)nc2ncccn2n1 C1(C(=O)NC(C2CCCN(CC(=O)NC3CCC(C)CC3)C2)C)CCC(=O)NC1 c1(COC(C(c2cccc(Cl)c2)N(c2n(C(C)C)cnn2)C)=O)ccccc1Cl Cc1sc2ccccc2c1C(=O)NCCCN(C(=O)CC1(O)CC1)C(C)C c1(CC)ccccc1NC(CC1(OC)CN(C(c2cccc(CCF)c2)=O)C1)=O C1(C(N2CC(CN(C(c3cc(C)no3)=O)C)C2)=O)CNC(=O)CC1(C)C N1(CC(c2cncs2)=O)CCN2Cc3ccccc3CC2C1 N1(CC(ONC(c2ccc(=O)n(C)c2)=O)C)CCC2OCCCC2C1 C1(C(N(C2CCN(C(c3cc(O)cs3)=O)C2)C)=O)CCCN1C C(C(O)(CNC(=O)CCNC(=O)CNC(=O)C(C)(F)NC(C)=O)CO)OC Cc1noc(N)c1C(=O)NCC1CC(NC(c2cccc(OCC(F)F)n2)=O)C1 CC1CC(CNC(=O)C(C)(C)NC(C2OC3CCC2C3)=O)CC(C)C1 CCC(O)C(C)(C)C(=O)NCCOC1CCN(C(c2cccc(F)c2C)=O)CC1 c1(C(N2C(CN(C(c3cnc(Cl)[nH]3)=O)CC)CCC2)=O)cnc2c(c1)CCC2 c1(C(=O)NCC2CC(NC(COc3c(C(C)=O)scc3)=O)C2)cnn(C)c1F CC1(C#CC(=O)NCC2CCCC2NC(c2cc3ccsc3s2)=O)CCCO1 C(=O)(C1=NNC(=O)CC1)N(CCCNC(C1CC=CCC1)=O)CC c1(NC(N2CC(C3(C(=O)OC)CCC(O)CC3)C2)=O)ccc2oc(O)nc2n1 C1(C(=O)NN)C2CCCCC12.C1(N(C)C(c2coc(CC)n2)=O)CC2CCC1C2 C(=O)(C(C)(C)CO)N(CC(=O)NC1C(C)(C(C)C)C1)CC1CC1 C1(CNC(C2(SC)CCN(C(C3CN4CCC3C4)=O)C2)=O)CCC(=O)NC1C N1(C(c2ccc(Br)c(F)c2)C(=O)NCC(=C)C)CCCC2(CC1)CCN(C)CC2 C(=O)(C(C)(CC)CCC(C)C)N(C(CCC)C#N)C C1(C(N2CC(NC(CSc3n(C)ncc3)=O)C2)=O)CCCN(c2cccs2)C1 CCCC(CC(=O)N1CC2CC1(C(=O)OC)C2)NC(=O)C(C)N(C)C N1(C(C(C)OC(C)(C)C)=O)CC2(CCCCN(C(=O)C=CBr)C2)C1 C1(CNC(C=CCCC)=O)CCN(C(C2CCC(CCC)CC2)=O)C(C)C1 C1(CNC(CCN(CC)CC)=O)CCCCN(C(C2CCN(OC)CC2)=O)C1 c1(CNC(=O)NC2CC(c3ccccc3)(CN)C2)ccc2c(c1)CNCC2 CCCCCCC(C)CC(=O)NCC1(NC(c2cscn2)=O)CC2CCC1CC2 N1(C(CC(C=C)C)=O)CCCC(CO)(CNC(=O)Cc2ccccc2C)C1 c1(OC)cccc(CC(=O)NC(C)C(C)NC(c2c(C(C)C)n[nH]c2C)=O)c1F C1(CC(=O)N(C(C)CC(F)(F)F)C)(NC(C(C)N2CCCC2)=O)CCCCC1 c1(-n2c(C(C)S(C)=O)nc(C(C)C)n2)ccccc1S(N)(=O)=O C(F)(F)(CN=c1nc2c(cnn2C)c(NCc2ccnc(Cl)c2)[nH]1)C1CC(C)C1 CCC(CC(=O)OC(C)(C)C)NCc1c(C)cnn1C1CCCCO1 C#CCC(C)(C)C(=O)NCC12CCC1CN(C(=O)C(c1cccc(Cl)c1)O)C2 CCC(C)(COC)C(=O)NCC1CN(C(=O)CCc2cc(C)on2)CCN1C N1(CC(=O)NC(C)C(C)NC(C2CCC(C(F)(F)F)C2)=O)CCCNS1(=O)=O c1(SC)ccc(C)c(C(=O)N(C)CC2CCCN(C(=O)Cc3c[nH]nc3C)C2)c1 CC(CC(=O)NCC(Cc1ccccc1)NC(C1CC(C)(O)C1)=O)NC(N)=O C1(C(=O)NC2CCC(C(N(OC)CC3CCCCC3)=O)C2)CCCCC(=O)N1 C1(C(=O)NC2CC(CNC(C3CCN(C(=O)OC)CC3)=O)C2)CC(=O)NC1(C)C N1(C(c2cc(C)c(F)cc2)=O)CCN(C(=O)Cc2c[nH]nc2O)C(C)C1C c1(CNC(c2c(NCCCOC)cccc2)=O)ccc(OC)c(C)c1C c1(CCC(=O)OC(C(=O)OC)(C)Cc2ccccn2)nc2ccccc2oc1=O C1(CNC(c2cc(OC(C)C)ncc2)=O)COCCN(Cc2cscc2Br)C1 CCC(CC)(CCN(C)C(c1cc(O)cs1)=O)NC(C1(COC)CC1)=O CCC(CC)(CCNC(=O)CNC(C1CC1C)=O)NC(=O)CCC1CC1.C(C)(OC)OC Cc1ccc(C(=O)OCCOC(=O)C(C)NC(c2ccccc2)=O)n1C C1(C(N(C2CSC2)CC#C)=O)CC(O)C(O)CC1CNC(c1ccc(C)cc1O)=O c1(OC)ccc(C(=O)NC2CCCCN(C(c3ccns3)=O)C2)c(OC)c1Cl c1(C(=O)NCC2CN(C(C3CC4CCC3O4)=O)CC2O)cc2cccnn2n1 Cc1cc(C(=O)NCCOC2CCN(C(=O)C(O)CC3CCCCC3)C2)co1 N1(C(C2CC3CC2CC3O)=O)CC=C(C(=O)N2CCOCC3(CC3)C2)CC1 C1(NC(C(CC)OCC)=O)CCC2(CC1)CCN(C(c1cc3occc3s1)=O)C2 N1(C(c2n[nH]cc2CNC(C2(C3CC3)CC=CC2)=O)=O)CCC2C(=O)NCC2C1 N1(C(c2cc(C)ns2)=O)CCN(C(=O)CCc2ccc(F)cc2)C(C2CC2)C1 O=C1COc2ccc(NC(N3CC4CC3CC4CN3CCCC3)=O)cc2N1 C1(C(=O)NC(CC)CNC(C2(CC)CC2)=O)COC2COCC12 N1(C(=O)NCc2cc(SC)nn2C)Cc2ccnn2CC1C c1(SCC(N2CC3C(NC(C=CC)=O)C(CC3)C2)=O)ccc([N+](=O)[O-])cc1 C1(F)(C(=O)NC(CNC(CCSCCCC)=O)CC(C)C)CC12CCCCC2 CC1C(C(=O)NCC2(O)CN(C(=O)Cc3nc(=N)[nH][nH]3)C2)=NOC1C c1(C(=O)NCC2(NC(C(CC#C)C3CC3)=O)CC2)[nH]c2ccccc2c1Cl c1(C(=O)NC2CN(C(CCc3c(C)n[nH]c3C)=O)C2)c(F)ccc2occc12 CC1(C(=O)NC(c2ccc(O)cc2)C(F)(F)F)CCCCNC1=O c1(C(=O)NC2CC(N(C(Cn3c(C)ncc3)=O)C)C2)coc2c1C(=O)NCCC2 N1(C(CSc2ccc(OC)cc2)=O)CCCC2(NC(=O)C3=CC4CCCC34)CC2C1 C1(CCOC)CN(C(=O)Cc2cn[nH]c2)CCN1C(c1cnc(C)n1C)=O C1(CC(N2C(C)(COC)CC2)=O)CN(C(c2cccnc2O)=O)CC1C C1(NC(N(c2ccc(OC)cc2)Cc2ccc(Br)cc2C)=N)CCn2ncnc2C1 C1(CC)CN(C(=O)NC2CCCCN2c2cc(OC)ncn2)CCO1 N#CC1(C(N2CCOC(CC(=O)Nc3cncc(F)c3)C2)=O)CCCC1 c1(N2C(C)CCC(NC(c3cncn(C)c3=O)=O)C2)ncnc2ccccc12 c1(C(=O)NC(CCCNC(CN(CC)CC)=O)C)cc(-c2cc[nH]n2)ccc1F C1(O)(CN(C)Cc2ncsc2-c2ccccc2)CCCC(C)(C)C1 N1(C(C23CC(C)(C2)OC3(C)C)=O)C2CCC1CN(C(C1CCS(=O)(=O)N1)=O)CC2 N1(C(CC=CC)=O)CC(NC(c2ccco2)=O)CC(C)(C)C1 C(C)(CCCCNC(C1CC1c1cccc(OC(F)F)c1)=O)NC(C=CCC)=O Cc1c(Cl)sc(Cl)c1C(N1CC(NC(C23CCCN2CCC3)=O)CC(O)C1)=O N1(C(CC(=O)N(C)C)=O)CCC(CCNC(C2CCC23CCC3)=O)C(F)(F)C1 C(=O)(C1Cc2ccc(F)cc21)N1C(C(C)NC(C2CCCC2C)=O)CCC1 c1(C(N2CCCC3CN(C(C(CC)O)=O)CC32)=O)sc2nc(C)nc(C)c2c1C c1(C(=O)NC2CN(C(c3c(C)cco3)=O)CC(C)(C)C2)coc2ccc(O)cc12 CCC(O)C(C)(C)C(=O)N1CCN(C(c2ccnc(O)c2)=O)C(CF)C1 C(=O)(C(C)(C)C(C)O)NC1CC(C)(CNC(c2c(C)cnn2C(C)C)=O)C1 C(=O)(C1=CC2CCCC12)NCCC1N(C(CC2C(C)(C)CCCO2)=O)CCSC1 N1(C(c2cccc(SC)c2)=O)CCC2CN(C(C3(O)CCC3)=O)CCC2C1 c1(CNC(C(c2ccco2)NC(C2OC3CCC2C3)=O)=O)cnc2n1CCC2 c1(C(N2CCN(Cc3ncn(C)c3)C3C2C3)=O)cccc(S(C)(=O)=O)c1 CC1OC(C)(C)OC1(C)c1nc(Cc2n[nH]c(-c3ccc(Br)cc3)n2)no1 c1(C(=O)NCCOCCCNC2CCC23CNC3)cc([N+](=O)[O-])cs1 C1(C(N2C(CNC(Cc3ccc(CC)cc3)=O)C=CC2)=O)CC2C(C1)C2(C)C c1(C(=O)NC2C(CNC(c3on(C)c(=O)c3)=O)CCC2)cccc2oc(=N)[nH]c12 c1(CS(N)(=O)=O)cccc(S(=O)(=O)NC(C2CCCCC2)CN(C)C)c1 N1(C(CCC(C)NC(c2occ3c2CCC3)=O)=O)CC(O)CC12CCC2 C1(C2(O)CCNCC2)(C(=O)NC(C(=O)OC)C)CCC1 c1(C(=O)NC(CNC(c2n(CC)ncc2)=O)CO)cccc(C#CC2CC2)c1 C1(NC(c2cc(S(N)(=O)=O)sc2Cl)=O)CCOc2cc(Br)ccc2C1 c1(C(C)=O)ccc(N(C(=O)C(=Cc2ccc(OC(F)(F)F)cc2)C)CC)c(F)c1 N1(C(c2c(COC)cco2)=O)CC2CC2C1NC(C1CC=CCC1C(F)(F)F)=O C1(C(N2CC(C)OCC2)=O)Cc2ccccc2CN1C(=O)Cc1cccc(O)c1 c1(NC(C(c2sccc2Br)NC(=O)OC(C)(C)C)=O)ccccc1SC1CC1 N1(C(CSS(C)(=O)=O)=O)CC2CC1(CNC(c1ccn(C3CCOCC3)n1)=O)C2 Cn1cnc2sc(C(=O)NCC(CNC(=O)Cn3cnc(=N)[nH]3)C(F)(F)F)cc12 CC1CCN(C(c2cc(Cl)sc2Cl)=O)CC1CNC(=O)CCC(C)(F)F c1(CC)cccc(F)c1C(=O)N(CC(C)NC(C1C(C(=O)OC)C1(C)C)=O)CC c1(OC)cccc(C(N2CC(CNC(C3(F)CCC3)=O)C(F)(F)C2)=O)c1C N1(Cc2cncc(C)n2)CC2CCN(C(=O)Cc3cc(Br)ncc3F)C2C1 C1(C(N(CCOC)CCNC(=O)CC=CC(C)(C)C)=O)CC(C)=NO1 N1(C(C(C)(C2CCC2)OC)=O)CCN(C(=O)CC2CCCC(OC)C2)CC1C N1(C(c2nccc(C)n2)=O)CCC2C(CCCN2C(c2cn(C)ccc2=O)=O)C1 C1(C(=O)NCC23CC(NC(c4ccc(C)cc4)=O)(C2)C3)(CC)CC(F)(F)C1 Cc1noc(C(C)C)c1C(N1CCC(C(C)NC(=O)Cn2cccn2)C1)=O CC1CC(=O)NCC1C(N1CC(=C(F)CNC(C2CC(F)C2)=O)C1)=O c1(Cn2ncc(CC(=O)NC(CC)C)c2)ccc(CN)cc1 C(=O)(CCC(C)(C)O)N(C(=O)CN1C(C)CCC1C)CCOC.C1(O)CC(CO)C1 CC1=C(C(=O)NCC2(C(=O)NCC3CCCO3)CCC2)Cn2ncnc2N1C N1(C(C2(C)CC3CC3C2)=O)CCN(C(c2ccccc2C2CC2)=O)CC(O)C1 Cc1nn(CC(F)F)cc1C(=O)NC1CCCN(Cc2ccc(F)cn2)C1 c1(C(=O)NCC2N(C(c3c(C)cc(C)nc3O)=O)CC2)c(C)c(C)cc(C)c1C C1(F)(CNC(C2(C)ON=C(C)C2)=O)CCCN(C(=O)CC2CC3(CCC3)C2)C1 CCCC(C)(CCC)C(=O)NCC1CCCCC1C(=O)NCc1ncnn1C CCC1=NOC(C(N2CCCC2CNC(c2cncc(O)c2)=O)=O)C1 C1(C(=O)NC2CC(C)(NC(C3CC3(F)F)=O)C2)CCC(C2CCCO2)O1 C(=O)(CCCCCCS(N)(=O)=O)N(CCC(C)NC(C1CSCCS1)=O)C C(CCC(=O)N(CCCNC(=O)COC(C)CC(C)C)CC)=CC C=C(CNC(c1cnn(C(C)(C)C)c1)=O)CCNC(=O)CC1OCCC1C N1(C(c2c(CC)ncs2)=O)CC2CCCC2(NC(C2SCC=C2C)=O)C1 N1(C(C(C)C2CCC2)=O)CC2CC1CN2C(c1cn(CC(F)(F)F)nn1)=O N1(C(c2ncc(CC)[nH]2)C(=O)NC)CCN(C(C)CCSC)CC1 c1(C(C)C)noc(C2CC2C(=O)NCCC(F)Cn2cc(C3CCCC3)nn2)n1 C1(NC(C=CCOC)=O)CCN(C(=O)Cc2ccc3c[nH]nc3c2)C12CCCC2 c1(C(=O)NC(CNC(C(CN(C)C)O)=O)C2CC2)cnc2[nH]nc(O)c2c1 C=CC(CC)C(=O)N1CC(C)(OCC(=O)NC2(c3ccccn3)CC2)C1 C=CC(C)(C)CC(=O)NCCCCC(N1CCCCC(COC)C1)=O C1(C(=O)Nc2ccc(NC(C(C)C)=O)cc2)CCCC2(CNC(=O)C2)C1 c1(C(=O)NC2(CC#C)CCC2)cccnc1CNC(C1CC12CC2)=O C1(NC(C(N2CCC(O)(CN(C)C(C3CC3)=O)C2)=O)=O)COC(C)(C)CO1 N1(C(C(N)c2cnn[nH]2)=O)CCN(c2cccnc2)C(=O)C1 C1(OCC2CN(C(C3(C)CC3)=O)C2)CC2(CCN(C(c3cccnc3)=O)CC2)C1 c1(CN(C(=O)CC2(CO)CC2)C)cccc(CNC(=O)C=CC2CCOC2)c1 CC(=O)CCN=C(NCc1ccc(Cl)s1)N(C)Cc1cc(F)ccc1F N1(C(CSCC#C)=O)C2CC=C(C(=O)NCc3cc(Cl)ccn3)C1CC2 c1(C2N(CC(N)=O)CCC2)ccc(Br)c(Cl)c1 C1(C(N(CCC(F)(F)F)C)=O)(NC(=O)CC2CC=CCN2C)CCC(C)(C)C1 c1(CNCCC23C(CN(C(=O)OC(C)(C)C)C2)C3)cnn2ncccc12 c1(OC)ccc(CCC(=O)NCC23CC(NC(=O)CSC)(CO2)C3)cn1 N(C1=NCCCNC(=O)N2CCC(N1)CC2)C1C(C(=O)OC)C1.C(C)(C)(C)O C1(NC(C(CCCC)N(C)C)=O)CC2CCC(C1)N2C(c1ccc(N(C)C)cn1)=O c1(CNC(=O)C(C2CC=CCC2)(CC)OC)ccc(CNC(=O)C(O)c2ccsc2)cc1 C(C(F)CCNC(C1(n2ccc(C(C)C)n2)CC1)=O)NC(CNC(=O)OC)=O C(=O)(C1CCCc2c(O)cccc21)NC(C)(C)CCCNC(c1ccc[nH]1)=O N1(C(C(=O)NCc2ccc(C#C)nc2)=O)CC2CN(C)CC2C1 CCCC(C(=O)NCC(O)CCNC(c1sc(Cl)c(Cl)c1C)=O)C(C)C CC1(C)C(NC(c2c[nH]nc2C(N)=O)=O)CC1C(N1CCCC1(C)C1CCC1)=O C1(NC(c2c(SCC)cccc2)=O)CCN(C(=O)C(Br)=C(C)C)CC1C C1(C)(C(=O)NC2C(CNC(c3c(-c4cn(CC)nc4)n[nH]c3)=O)C2)CNC(=O)C1 N1(C(C2CC(C)C2)=O)CC2CC2(CNC(c2ncoc2-c2ccccc2)=O)C1 C1(C(=O)NC2CC(C)(NC(C=C3CCN(C)C3)=O)C2)CCC(F)(F)C1O c1(C(=O)NC2CC3(C(NC(=O)CO)C3)C2)[nH]c2ccccc2c1Cl Cc1cc(NC(=O)C(=O)NCC2=NOCC2)c2occc2c1 N1(C(C2(COCC)CC2)=O)CC2(CCC2)CC1C(=O)N(CC(C)(C)C)C c1(C(=O)NC2CN(C(C3(CC#C)CCCO3)=O)CC2O)c(C)oc(C)c1C N1(C(c2c(CC)csc2)=O)CC2(CC(C(=O)NC(C)CC(C)O)CO2)C1 C1(O)(CN(C(C(C=C)O)=O)C)CCN(C(=O)C(C#N)C2CC2)CC1 N1(C(c2ccc(CCCC)cc2)=O)CC2(CNC(=O)CNC(=O)NC)CC1CO2 c1(C(N(C(CNC(C(COCC=C)c2ccccc2)=O)C)C)=O)ncccc1F c1(C(N(CCNC(CCC=C(C)C)=O)C2CC2)=O)cc(OC(F)F)cc(OC)c1 C1(CCOC)CN(C(C2(CCO)CC2)=O)CCN1C(c1cn(CC(F)F)cn1)=O N1(C(CC2N(C(CCn3ccc(C)n3)=O)CC(F)C2)=O)CCC2(CNC(=O)N2)C1 c1(OCCC#C)ccc(C(N2CC(F)CC2CN(C)C(C2(C)CC2C)=O)=O)cc1 N1(C(c2n(C)ncc2)=O)C(C(=O)NC2(n3cccc3)CC2)C2(CC2)C1 C=CCC(C)(CC)C(=O)N(CC(C)NC(=O)CN(C(=O)C(C)C)C)CC c1(OC)ccc(CNCCNc2ccc(C)n2Cc2ccccc2)cc1Cl C1(C(=O)NCC(C(C)(F)F)Cl)C2CC3C(C2NC(=O)Cc2ccc(O)cn2)C13 C1(NC(=O)CSC(F)F)CC2CCC1CC2NC(c1ccc(O)c(Cl)c1)=O C#Cc1ccnc(C(=O)NCC(O)CN(C)C(c2sccc2C2CC2)=O)c1 c1(NC)cncc(C(N2CC(NC(=O)CC3CC(=O)NC3=O)C(F)C2)=O)c1 c1(C(N2CCC3(CCCC3C(N3CC(F)(F)C3)=O)C2)=O)cncc2ccccc12 n1(CC)ncc(Cl)c1C(N1CC(OC)C(NC(c2cccc(C)c2)=O)C1)=O N1(C(CC2CC(OC)C2)=O)CCCC(N(C)C(c2ccsc2C)=O)C1 CN1c2ccccc2N(C(c2cscc2Cl)C(=O)NC2CC2)C2(CC2)C1 C1(N(C(CC=C)=O)C2CC2)C2CCC1CN(C(=O)CCSc1ccc(F)c(F)c1)C2 c1(C(=O)NC2CC2CNC(C23CC(O)C2C3)=O)ccc(-n2ccnn2)cc1 c1(C(=O)NCC2N(C(C(C)SC)=O)CC=C2)c(O)nnc2c1COCC2 CC(C)CC(C)OCC(=O)NC(C)(C)CNC(=O)CCC1(C)CC1.C(N)(=O)N N1(c2ncc(CC)cn2)CCCC(C(=O)N(CC)CC2CC23CCOCC3)CC1 Cc1nc(C)c(C(N2CCCC2C(C)(C)NC(=O)CC2CC(C)OC2C)=O)s1 c1(C(N2CCC3(C(C(N4C(C)C(=O)NCC4)=O)C3)C2)=O)ccc2cncn2c1 N1(C(C(CC#C)(C)C)=O)CC2CCC1C(CNC(c1ccc(Cl)c(C#N)c1)=O)C2 c1(C(N2CCC(NC(c3coc(Cl)c3)=O)C2)=O)cc2ncccc2cc1Cl C1(CNC(C2C(OC)C2)=O)CCN1C(=O)CCC1CC1(C)C C=CCC(CNC(c1cnn(C(C)C)n1)=O)NC(C1CC1C(C)C)=O c1(C(=O)NC(CC)CNC(C2CC3(CSC3)C2)=O)cnc2scc(C)n2c1=O Cc1cccc2cc(C(=O)NC(C3CCCN3C(=O)C(C)C(F)(F)F)C)cnc12 N1(C(c2ccc(CC)s2)=O)CCN(C(C)CNC(=O)Cc2ccc(F)cc2)CC1 C1(C(=O)NCC=C)CC=CCN1C(=O)CCC1(CCCC)CCCC1 Cc1cc(C)c2cc(C(=O)NC(C)CC(C)NC(=O)Cc3ccoc3C)[nH]c2c1 N1(Cc2ccc(NCc3cccc(OC)c3)cc2)CCCC2(CC=CCO2)CC1 C1(NC(C(C)=C2CCC2)=O)CCN(C(=O)C(=O)C(F)(F)F)C12CCC2 C1(NC(COC(C)C)=O)CCOCC1NC(=O)CCC12CCC(CC1)C2 N1(C(c2nccc(CC)c2)=O)CC(C)C(NC(c2cocc2C)=O)C(C)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(CNC(=O)Cc2nccn2C)C(C(F)(F)F)C1 N1(C(CN(c2ccncc2)C)=O)CCN(C(=O)CC2CC=CCC2)C(C(F)F)C1 c1(C(N2C(c3cccc(OC)c3)COCCC2)=O)cnc(O)c2cncn12 c1(C(C(=O)N(CC(C)NC(C(CC)=CC)=O)C)C)ccc(C#N)cc1 c1(CN(CC(=O)NCC(C)CNC(=O)CN(C)C)C)c(Cl)cccc1Cl C(CCCC(C)NC(c1conc1C1CCC1)=O)NC(c1cc(CC)no1)=O C1(CNCC=C2CCN(C(C(C)(C)c3cnsc3)=O)CC2)CC(C)(C)C(=O)N1 c1(C(=O)NC(C(=O)NC(CC=C)CC(F)F)c2ccoc2)ccn2ccnc2c1 c1(C(=O)NC2(CNC(c3c(C(C)(C)C)n[nH]c3)=O)CC2)cc2cc(F)ccc2[nH]1 c1(-c2cc(C(N(C3CCC(NC(C4CC(=C)C4)=O)C3)C)=O)sc2)ccc(F)cc1 C1(NC(N2CC(C)(OC)C2)=O)CS(=O)(=O)CC1C(N)=O C1(C(=O)NCCc2cc(C)ncc2)CN(C)CCN1C(=O)CCC1CCOCC1 c1(CNC(c2ccccc2F)C)cc2ccccc2c([N+](=O)[O-])n1 C1(=O)C2CCCNN=CC=C2CN1.N1(CC(=O)OC)CC(C)(C(=O)OC(C)(C)C)C1 c1(CNC(C2C(CNC(c3ccc(C#C)o3)=O)OCC2)=O)ccc(C)c(O)n1 C#CC1(NC(C2(NC(=O)C=CCO)CC(F)C2)=O)CCOC1 C(=O)(C(F)(F)C(F)(F)C(F)F)N(CC(CC)NC(c1c(CC)cc(F)cc1)=O)C c1(CC(=O)NC(C)C(CO)NC(=O)CSC2CCCCO2)c(Br)cnn1C C1(NC(C(C)NC(C)=O)=O)CC(F)(F)CC1NC(=O)CC1(C)OCCO1 CCC(O)(CC)CCNC(=O)C=CC1CCCN1C(c1cnn(C(F)F)c1)=O C1(CNC(CC=CC=C)=O)CC2CN(C(C3CC3c3ccc(C)s3)=O)CC12 N(C1CCCc2c1cnn2CC(=O)OC)C(CCCC)CCO c1(C(=O)NCCC2CN(C(C(CCC)(C)CC)=O)C2)n[nH]c2ccc(OC)cc12 N1(C(C(F)=CCC)=O)CC(C2CCN(C(=O)Cc3ccc(O)c(C)c3)CC2)C1 N1(C(C2CC(N(C)CC)C2)=O)CCC2(CC(C(=O)N(CCN=[N+]=[N-])C)C2)C1 CCC(C)(C(=O)N1CCC(CCNC(c2coc(COC(C)(C)C)n2)=O)C1)OC C1(NC(C(C)OCCC(C)C)=O)CCCC1C(=O)NCC(C)(O)CO C(=O)(CC1CCCc2c(O)cccc21)N1C2C(NC(c3ccccc3)=O)C(C2)C1 c1(C(=O)NC2CN(C(Cn3c(C(C)C)ncc3)=O)C3C2C3)cc(F)cc(N)c1F N1(C(C2(COC)CCC2)=O)CCC(C(F)(F)F)C(NC(=O)C=CC=C(Cl)Cl)C1 c12ccc(cc1)NC(=O)N2.c1(NCCCC2CCOC2)nccc(CO)n1.C(F)(F)F C(=O)(C1OCCc2c(O)cccc21)NC(CCN(C(CCC=C)=O)C)C(C)C c1(CCC(=O)NC2CC(N(C(C3C(C(=O)OC)CC3)=O)C)C2)ccc(F)cc1 c1(CNC(C2C(NC(c3nccs3)=O)C2)=O)csc(Br)c1 N1(C(C(C)N2CCC2)=O)CC2CCCC1C2CNC(c1ncccc1Cl)=O C(=O)(C1CCc2c[nH]nc21)N1CCC(NC(C(n2ccc(C)n2)C)=O)C(F)C1 N1(C(CC(C)CF)=O)CCC2(CCOCC2)C(CNC(=O)CNc2nccs2)C1 n1(C(C)C(=O)N(C2(CO)CCSC2)C)cnc(C#N)n1 c1(C(N(C)CCN(C)CCc2ccccc2)=O)ccccc1 C12(CCC(=O)NCCc3cc(C)[nH]n3)CCC1CN(C(=O)C(C)SC(C)C)C2 CC1CCC(NC(c2cnc(S)n2C2CC2)=O)CN1C(c1cnn(C)c1)=O Cc1ccc(F)c(C(=O)NCCCC(C)NC(=O)CC2CC(F)(F)C2)c1F CN1CCCCC1C(N1CCCC(CCNC(=O)CCCN2CCCCC2)C1)=O Cc1[nH]c(=N)sc1C(=O)N(C)CCNC(C1(n2cncn2)CC1)=O N1(S(CC(=O)OC)(=O)=O)CCCCC(CC(=O)NC2COC(C)C2)C1 c1(C(N2CC(N3CCNC3=O)C2)=O)cccc(CO)n1.N#CC1CC(N2CC2=O)C1 N1(C(C(CC(C)C)O)=O)CCC2CN(C(c3ccc(-c4ccco4)s3)=O)CC2C1 C(=O)(CC(C)(C)CC(F)(F)F)NCC(C)(C)CCNC1N(C(C)=O)CCC1 c1(CCC(C)C)ccc(CN(C(=O)C(=O)NC2CCCC2CN)C)cc1 C1(C(N(CC(F)F)CCC)=O)CCCN1NC(=O)C=Cc1ccnn1C CC(C)CCC(=O)C(=O)NC(C)CC(C)NC(C1CCCC(C)CC1)=O N1(C(C=CC(C)(C)SC)=O)CC2CCC2(CCNC(c2nc(C)ccc2F)=O)C1 Cc1noc(C)c1CCC(N1CCC(C)(CNC(=O)Cc2ccnc(F)c2)C1)=O CC(CCC(=O)NCC1CC(C#N)C1)NC(=O)CCc1nccn1C C12(C(N(CCCCN(C)C(C3COC(=O)O3)=O)C)=O)COCC1C2(F)F n1(CC)cc(Br)cc1C(=O)NC1CN(C(=O)CCn2c(C)ccc2C)C1 Cn1c(C(N2CC3CC(NC(c4ccc(F)cn4)=O)C2C3)=O)cc2ccccc12 c1(C(=O)NCCN(C(Cc2ccc(OC)nc2)=O)CC2CC2)c[nH]cc(Cl)c1=O C(=O)(C#CC1(C)CCCO1)NCC(CNC(c1c(F)ccc(C)c1)=O)CO Cn1nncc1NC(=O)CC1(C)CCN1C(c1ccon1)=O C(=O)(CC(C)(C)C#N)N1CCCC(C(C)NC(Cc2c(C)noc2C)=O)C1 N1(C(COCCOCC#C)=O)CC2CCN(C(c3ccc(F)c(C)c3)=O)CC12 O=C(C(F)(F)C(O)c1ccccc1)Nc1ccc(N2CCC(CO)CC2)nc1 C(C(=O)NC(C)(C)CC)(C(C)CC1CC1)N1CCN(C(CC)(C)C)CC1 N1(C(CCC)=O)CCCN(C(c2ccc(N(C(=O)CC)C)cc2)=O)CCC1 C1(C(N(C(C)CCNC(c2coc(C(F)(F)F)c2)=O)C)=O)CCCC2(CCC2)C1 N1(C(C(C)(CO)NC(CC(C)(C)OC)=O)=O)CCC(O)C(C)C1 N(C1CCCc2c[nH]nc21)C(C1N(C(CCSCCCC)=O)CC(O)C1)=O Cc1noc2cc(C(=O)NCC(O)CCNC(=O)CS(=O)(=O)N(C)C)ccc12 N1(C(C(C)=O)=O)CCCCC1C1CN(C(C2CC2C2CC2)=O)C1 c1(C(N)=O)ccccc1S(=O)(=O)N1CC(CC(F)F)C1 O=C1OCC2CN(C(N(CC3CCC3)CC3CC3)=O)CCC12 N1(CCC)CC(CNCC2CCOCC2OC)CC1=O CC1CC(NC(=O)Nc2ccc(SCCC(N)=O)cc2)CC12CCC2 c1(CCC)n[nH]c(=NCC2(CCN(C(=O)C(O)CC(C)C)CC)CC2)s1 c1(C(=O)NC2CCC(NC(C3(COC)CC=CC3)=O)C2)coc2ccc(O)cc12 C(=O)(CC1=CCN(C)CC1)NC(C1CCN(C(=O)OC(C)(C)C)C1)C C1(N(C(=O)C=CC=C(Cl)Cl)C)CCCC(N(C)C(c2nonc2N)=O)C1 c1(C(N2CCC(CF)C2)C(=O)NC(C2CCC(C)(C)C2)=O)cccc(N(C)C)n1 c1(C(=O)NCC(CC=C)C(=O)N2CCCOC(C)C2)cccc2[nH]ccc12 C1(NC(Cc2nc(C)c(C)o2)=O)CCCN(C(=O)CCOC(C)C)CC1 C1(C(=O)NCC2C(CNC(C(CSC)O)=O)C2(F)F)CCn2nccc2C1 C#Cc1ccc(C(N2CC(CNC(C3CC(CCO)C3)=O)C(C)C2)=O)cc1 c1(C(=O)NCC2(CNC(c3c(C)sc(O)n3)=O)CCCC2)c(O)cccc1F C1(C(N2CCC(=CCNC(CCC(C)OCC)=O)CC2)=O)CC2(C1)CC(F)C2 N1(C(C)=O)CCOCC1C(=O)NCC1CCN1C(=O)CCSc1nnnn1C N1(C(C(CC)OC)=O)CCN(C(c2cnccc2N(C)C)=O)CCC1C C1(n2cc(-c3ccc(OC)cn3)nn2)CC2CCC1(C(=O)NCc1ccon1)C2 C(=O)(CCCCCCCBr)NC12C(CN(C(CC=C)=O)C1)CCC2 c1(C(=O)NC2CC3(CN(C(CC(C(CC)C)O)=O)C3)C2)ccn2ncc(C)c2n1 C1(NC(=O)Cc2nc[nH]n2)CC2(C1)CN(C(=O)C(F)CC1CCCC1)C2 N1(C(c2nc(CC)sc2)=O)CCC(C)C1CNC(c1cnc(C2CCCO2)s1)=O Cc1nc(-c2ccccc2)[nH]c1C(=O)NCCCCCNC(C12CC(C)C1C2)=O Cc1coc(C(=O)NCCC(C)(C)NC(c2coc(Cn3cccn3)c2)=O)c1 c1(C(N2CC(N(C(CCCOCCC)=O)C)C(O)C2)=O)cnc(C)nc1C C#Cc1ccc(CC(=O)NC2(CCO)CN(C(=O)OCC)C2)cc1.C(C)(C)(C)O c1(C(N2CCN(C(=O)C(F)C3CCOC3)CC2)=O)cc(Cl)c2c(c1)OCCO2 N1(c2snc(COC)n2)CCC2(NC(=O)C(C(C)CC)OC)CCCCCC12 CC(C)CCCC(=O)N1CC2C(c3cn(C4CCC(=O)N4C)nn3)C2C1 c1(N(C)CC2CCCC2O)nc(N(C)Cc2nnc3n2CCC3)c2ccsc2n1 N1(C(c2ccc(C)nn2)=O)CC(NC(C2(C)CC=CCC2)=O)CC(F)(F)C1 N1(C(C(=O)NCCC)CC2CCC(C)(C)O2)CCCOc2ccc(C)cc21 N1(C(c2cc(C(C)=O)on2)=O)CC=C(CNC(c2cc(C)cc(C)n2)=O)CC1 C1(C(N(CCC=C)CC)=O)CC12CCN(C(c1c(OC)ccc(Cl)c1Cl)=O)CC2 Cc1cc(C#N)ccc1C(N1CCC(NC(=O)CSCCN(C)C)C1)=O N1(C(CCNC(c2coc(CO)c2)=O)=O)CCOC2CCCCC12 C1(CCCCNC(CCC)=O)CCCN(C(=O)C(c2ccc(Cl)cc2)C)C1 c1(C(N(CC(C)NC(Cn2nc(C)c(C)c2C)=O)C)=O)cccc([N+](=O)[O-])c1 N1(C(C(C)OC)=O)CCCCC1CCNC(=O)CC(O)c1ccccc1 N1(C(Cc2c(C)scc2)=O)CCCOC(CCNC(c2ccc(Cl)cc2F)=O)C1 C1(CCC)(C(=O)N(C)CCNC(C2CC(OC)C(OC)C2)=O)CCNC1=O N1(C(C2C(=C)C2)=O)CCCC2CN(C(c3cc4c[nH]nc4s3)=O)CC12 CCC(C)C(O)C(C)C(=O)N1CCC(c2cccc(F)c2)C1 C1(CNC(=NCc2ccc(SC)nc2)NCC(F)F)CCC(=O)N(C)C1 c1(OC)cnc(C(N2CCCC(O)(C(=O)Nc3cc(O)ccn3)C2)=O)c(F)c1 N1(C(C(=O)NCC(C)C)CC(C)SC)CC2CCC(C1)N2c1ccccc1 c1(OC)nc(C)ccc1C(=O)N(CCNC(c1ccon1)=O)Cc1ccccc1 c1(OC)c(CCNc2cccc(CN3CCCC3=O)c2)cccc1O C(=O)(CC(O)C(C)C)NCC1(C(=O)NCc2ccc(OC)nc2)CCCO1 c1(OCC)ccccc1C(=O)NCC(O)CN(C(=O)CC1CC1(C)C)C C(C(C)(O)CC(=O)N1CC(O)CCC1C(=O)NCC1(O)CC(O)C1)OC N1(C(=O)C=Cc2cccnc2)CCC2(CCN(C(c3cnccn3)=O)CC2)C1 C1(ONC(Cn2cc(NC(CCCn3c(C)ncc3)=O)nn2)=O)CCS(=O)(=O)C1 Cc1ccc(C)c(OC2CN(C(=O)CC3(OCc4ccccc4)CC3)C2)c1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC2CC(C1)CN(C(c1ccco1)=O)C2 C1(C(=O)NC(CC(=O)N2CC(COC)C2)COC)CCC(O)CN1C CC(CCCC(=O)OC1CCC(O)C1O)Oc1csc(C(C)(F)F)n1 CC(=Cn1ccnn1)C(=O)NCC(CO)NC(=O)CCC1CC1CC1CC1 C1(C)(CNC(C(c2ccoc2)NC(Cc2cn(C)nc2)=O)=O)CCCCC1 CC1CC(CNC(C2(C(F)F)CCC2)=O)CN1C(C1CC12CCSCC2)=O C(=O)(CCCS(C)(=O)=O)NC(C1(O)CCN(C(CC(C)C(F)F)=O)CC1)C c1(CC(=O)NCc2ccc(C(=O)NCC(F)Cl)s2)cccnc1O C=C(CNC(c1ccncc1C)c1nnnn1C)c1cccc(F)c1 C(CCC(C(=O)NC1CC(=O)NC(=O)C1)NC(=O)Cc1c[nH]nc1O)OC C1(C(=O)NC2CN(C(CCNS(C)(=O)=O)=O)C2)CC12CCOC2 CC1(NC(C2CCC3CCC23)=O)CCN(C(=O)CSCc2ccncc2)CC1 c1(CNC2C(CC=C)CCC2)n[nH]c2ccncc12 C=CCC(F)(F)C(=O)N1CCC(CO)(NC(=O)CNC(c2ccc(F)cc2)=O)C1 C1(NC(c2c(C)oc(CO)c2)=O)CC(O)CN(C(=O)CCCc2cnn[nH]2)C1 C=Cn1nccc1C(=O)NCCC1(O)CCN(C(=O)CC2(OC)CCOCC2)C1 C1(C(N2CCCC(O)(CCNC(C34CC(CO3)C4)=O)C2)=O)CC2(COCCO2)C1 N1(C(C2C(OC(C)=O)C2)=O)C(CNC(C2CN(C)CCO2)=O)CC2CCCC12 C1(C)(C(N2CC(O)(C(C)NC(C3(OC)CCC3)=O)C2)=O)CCCS1(=O)=O C(CCCCC(=O)NCCCCCNC(C1(C)CCC(=O)N1)=O)SC C1(C2CC(c3onc(C)n3)C2)CC2(CCC(CN)OC2)C1 c1(OC)cc2c(cc1NC(CCc1nccs1)c1ccco1)OC(C)C2 C(c1ccc(Cl)s1)=CC(=O)N(CC(C)N(C)C(c1cnnc(O)c1)=O)C C1(C(C)NC(=O)COc2cnn(C)c2)CCCN1C(=O)CCC1CC1(F)F C(=O)(C1CCCc2nc[nH]c21)NC(C)CNC(=O)C(=O)NCC1CC1 c1(C(N2CCC(CNC(c3ccn(CC)c(=O)c3)=O)C2)=O)cc(Cl)cc(F)c1F n1(SCC)ncc(C(=O)NC2CCC(CCC(=O)CCc3cc(Cl)no3)C2)n1 C(=O)(C1=CCCOCC1)NC(C1CN(C(c2ccc(Cl)o2)=O)C1)C c1(-c2n(C3CCS(=O)(=O)C3)nc(CO)n2)ccc2cccc(Br)c2n1 C(=O)(C(C)(CC)CCC)N1CCC(=C)C(CO)C1.C12(CCC1)C(=O)NOC2=O C1(NC(C(CNC(c2cn(CC)nc2)=O)O)=O)CCS(=O)(=O)C1 C12(C(=O)NCC3CN(C(C4C(COC)C4)=O)C3)CCC(N=[N+]=[N-])(CC1)C2 c1(OCC)ccc2c(c1)nc(NC(=O)Nc1ccn3nccc3c1)n2C(F)F N1(C(C(C=C=C)C)=O)CCC2(CC1)CC2CNC(=O)N(C)C CCC(CC1CCCCC1)C(=O)N1CCC1CNC(=O)C(C)(C)NC(C)=O N1(C(CCC2CC(NC(=O)C(C3CCOCC3)=O)C2)=O)CCOC2CCCCC12 c1(C(=O)NCC2C(CNC(Cc3ccn(C)n3)=O)C2)cncc2ccsc12 c1(OC)ccc(-c2cnc(CNC(=O)CN3CCCC(N(C)C)C3)s2)c(C)c1 C12(N(C(CC(=C)C)=O)CCOc3ccccc3)CCC1CN(C(=O)CC(C)(C)C)C2 c12[nH]c(c(C)c1C)-c1ccccc1OC2=O.c1(N(CC=C)CC=C)nccs1 N1(C(Cc2cc(C)sc2C)=O)CCN(C(=O)CCC2CCCN2C)CC1CF C=CCCCC(C(=O)NC1CCCCC12CCC2)NC(=O)CC(=O)N(C)C C1(OC)CN(C(=NCCC(F)(F)F)NCC=O)CC1C(=O)OC(C)(C)C C1(C(N(C)Cc2cn(C)cn2)=O)CCC(C)(C)N(C(=O)C2=C(Cl)CC2)C1 C(CNC(c1csc(CNC(=O)CCC2OCCO2)c1)=O)(C(C)C)OC C1(C(N2CCCC(NC(c3cc(OC)n[nH]3)=O)CC2)=O)Cc2ccccc2CO1 C(=O)(C(CC=CC)NC(c1ncccn1)=O)NC(C#C)CC1CCC1 C(=O)(CC(O)C(C)CC)NC(C(=O)N1CC(SCC)C1)CC(F)F Cc1nc(C)c(C(=O)NCC(N2CCN(C(=O)CC3CCC(C)(C)C3)CC2)C)o1 N1(C(c2c(C)snc2)=O)CCCCC1CC(=O)NCCCC(C)O N1(C(=O)CCC2CCCCO2)CC2COCC2(C(=O)NCc2ncccc2O)C1 C(N=C(NCc1cccs1)NC(C1(C#N)CC1)C(F)F)c1ccc(SCC)o1 CC(C)(CN=c1[nH]c(NCC2CCCC2)nc2c1CCC2)c1cnc[nH]1 c1(C(=O)NC23CCN(C(C4CCC(OC)C4)=O)CC2C3)cc2cc(C)ccc2[nH]1 N1(C(c2n[nH]cc2F)=O)CCCN(C(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(C)(NC(=O)NC2CCC(=O)NC2=O)CC1 C1(N(C(=O)C(N2CCCCC2)=O)CC)C(C)OCC12CCNCC2 c1(C(N(C2CCCN(C(C3CSCCS3)=O)C2)C)=O)cn2c(n1)CCC2 C1(NC(C2N(CC)CCC2)=O)CC2CCC1C(NC(=O)CCc1ccncn1)C2 c1(C(N(CC(CC)(C)NC(=O)C(=O)NCC)C)=O)ccc(-n2ccnc2)c(C)c1 N1(C(C2CCN(C(C3C=C(C)CS3)=O)CC2C)=O)CC2CC(C1)N(C)C2 C1(C(=O)NCC23C(CN(C(C(CC)=CC)=O)C2)C3)CC2C=CCC(C1)C2 c1(N(C)Cc2cccc(N)c2)nc(N(C)CC2(F)CCCC2)nc2c1SCC2 C1(NC(CS(N)(=O)=O)=O)CS(=O)(=O)C12CCN(C(=O)Cc1nncs1)CC2 N1(C(C2C(C(C)(F)F)C2)=O)CCC(CO)(CNC(c2cccc(Cl)c2)=O)CC1 C(=O)(C(C(C)C(C)(C)C)N1CCCCCC(CN(C)C)C1)NCC(C)C N1(C(Cc2onc(C(C)C)n2)=O)CC2(CCC2NC(=O)C(C)c2cncs2)C1 C(C1=CCCN(C(=O)C2=COCCO2)C1)NC(C1(CC=C)CC1)=O Cc1cc(O)c(CN2CCNCC2C(=O)NCCCCCCO)cc1Cl Cc1ccc(C(N2CCC(NC(c3cc(Br)no3)=O)C(CO)CC2)=O)c(N)c1C N1(Cc2ccc(OCC(=O)NC)cc2O)CCC(F)(F)C(C(F)(F)F)C1 N1(C(Cc2nnc(C)s2)=O)CCCN(C(C2CCCN2CCC(C)C)=O)CC1C C1(N(CC(=O)Nc2nccn2C)C)CN(C(=O)C#CC2(C)CC2)CC1C1CC1 CC1(NC(c2cc(F)ccc2Br)=O)CCCN(C(C2CC3(CCC3)C2)=O)C1 C1(NC)CCCC(N(C)C(c2ccnc(-c3ccccn3)c2)=O)C1 c1(NC(=O)CC2CN(C(C3CCC(F)(F)C3)=O)CCO2)cnncc1Cl c1(C(=O)NCCN(C(c2c(CC)nns2)=O)C)cncc(O)c1Cl C1(NCC2CC(=O)N(C)C2)CN(C(c2nc(NC(C(C)C)=O)sc2)=O)CC1O N1(C(CC)=O)CCC2CCN(C(=O)Cc3cccc(Br)c3Cl)C2C1 C(C(CO)C(=O)NCCC(CNC(=O)CCC(=O)Nc1nccs1)OC)OC C1(CNC(C(C)(C)F)=O)CN(C(C2CCSC2)=O)CC1C(F)(F)F C(CC(=C)Cl)(C(=O)NC(C1CCC1)C1CCC1)NC(C(CC#C)O)=O N1(C(C2(CC=C)CCCC2)=O)CCC(C(=O)NC2CC(n3cncn3)C2)C(O)C1 C12(CNC(CC(C)OC)=O)CN(C(c3ccc4cnnn4c3)=O)CC1CCO2 N1(C(C)=O)CCN(C(=O)C(c2cnc(C)s2)N(C)C(C2(CO)CCCC2)=O)CC1 CC1CCN(C(=O)C(=O)Nc2ccc(-c3ccco3)nc2)CC1CO n1(CC(=O)NC2C(CNC(=O)C=C3CCC3)CCC2)[nH]cc2c(=O)ncnc1-2 c1(NC(C2(C)C=CCC2)=O)cccc(NC(C23CCC(CC2)O3)=O)c1 N1(C(Cn2ncc(C)c2)=O)CC(CNC(=O)Cc2ccn(C(F)F)n2)C(C)C1 c1(CC(N2CCC(C3N(C(C(F)=CC)=O)CCCC3)C2)=O)c(OC)cccc1C c1(OC)cc(C)cnc1C(=O)NC1CCN(C(c2ccc(F)cc2C(F)F)=O)C1 N1(C(C(CC)NC(N)=O)=O)C2CCC(C2)C1C(=O)NCCCC1(C)CC1 c1(OC)c(C(=O)NC2(CCC(=O)NCC3CC4C=CC3O4)CCC2)csc1Cl C(=O)(CC(CNC(C1CN2CCC1C2)=O)C1CCC1)Nc1c(C)csc1 C1(CC)CCCN(C(=O)CN2CC3CC3C2)C1.N1(CC(C)CO)CCCC1=O c1(CC)onc(C)c1C(c1nnnn1C1CCC1)NCC1CC(CF)C1 CCC(C(=O)N1CCC(CCNC(=O)C(=O)N(c2ncc[nH]2)C)CC1)C(C)O C(=O)(C(O)C(F)(F)F)NC(C(N1CCC(N(C)CCO)C1)=O)(C)C c1(SCC(NNC(c2c(C)cc(C(=O)OCC)nc2)=O)=O)c(C)nc(C)nc1O C(=O)(C(C)(C)C(=O)NCC(C)(C)NC(c1cc(Br)n(C)c1)=O)N(C)C C(C1CCc2nccn21)NC(C1CN(C(c2ccc[nH]2)=O)CC(C)O1)=O C(C)(C(=O)N(C)CC1(O)CCCN(C(=O)C(C)=C2CCC2)C1)(C(C)C)NC(C)=O Cc1csc(C(C)NC(=O)CN(C(=O)Cn2nccn2)C)n1 C(CCC1CC1)(C(=O)NCc1cc(Cl)ccn1)NC(CCNC(=O)NC)=O Cc1ccncc1C(=O)NC1CN(C(c2cc(C(N)=O)no2)=O)CC1F N1(C(c2cccc(OCC)n2)C(=O)NCC(C)C)CCC12CCCSC2 CC1=NOC2(C1)CC(C(=O)NCC1CC(NC(=O)Cc3cnoc3)C1)C2 N1(CCC(N2CC(OCCNC(C(C)(C)CF)=O)C2)=O)C(=O)NC(C)(C)C1=O c1(C(N2CC3C(CNC(CC4COCC(C)O4)=O)C3C2)=O)ccc(F)nc1F CC(C(CO)NC(=O)CNS(=O)(=O)C1CC1)NC(c1cnn(CC(F)F)c1)=O Cc1ccccc1C=CC(N1CC(O)CCC1C(=O)N(C(C)CC1CC1)C)=O C1(NC(C(N2CCOCC2)C)=O)CC12CC(C(=O)NCC13CC1CNC3=O)C2 N1(CC(=O)OC2CCCCCC2c2ccccc2)C(=O)c2ccccc2C1=O C(CCCCCNC(c1ncc(Cl)n1C)=O)NC(C(C)c1ccsc1)=O C1(NC(c2ccsc2Br)=O)(CO)CCN(C(C2NC(=O)C3CC23)=O)CC1 C(=O)(C(F)C(C)(F)F)N1C(C(C)NC(C2CCCS2)=O)CCC1 c1(C(N2C(CNC(C3C(C)CC=CC3)=O)CN(C)CC2)=O)cc2ccncc2[nH]1 CC1CC=C(C(=O)NCc2cccc(NC(c3ccc(O)c(Cl)n3)=O)c2)CC1 C12(CNC(c3c(C)n(C)cn3)=O)CCCC1CCN2C(=O)COc1ccn(C)n1 CC1CC(C(=O)NCC2(CNC(c3ccc(C(C)(F)F)nc3)=O)CC2)CC(C)C1 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCCC(O)(CNC(c2nn(C)cc2C)=O)CC1 C1(C(N2CCC(CC=C)(NC(=O)CC(C)F)C2)=O)CC(C(C)C)=NO1 n1(CC(=O)N(CCCNC(C2CC23CC3(F)F)=O)C2CC2)ncc(O)nc1=O c1(C(=O)NC2CN(C(C3(CF)CC3(F)F)=O)CC2F)ccc2ccsc2c1 C1(C)(C(N2CCC(C)(OC)CC2)=O)Cc2ccccc2C1 n1(CC)cc(-c2n[nH]cc2C(=O)NC2CC2NC(C2CC(N(C)C)C2)=O)cn1 N1(C(c2c(C)cc(C)o2)=O)CCN(C(c2ccccn2)=O)C2COCC12 CC1CCN(CC(=O)NCCCC(CO)NC(C2CCNC(=O)C2)=O)CC1 C(=O)(CCCC(C)(C)C)NCC1N(C(C2=CC(C)(CC)C2)=O)CCC1 C=CC1CCN(C(C2CC3CC3N2C(=O)CCNC(=O)OC)=O)CC1 C=CCC(CC)C(=O)N1CCOCC1C(=O)NCC(n1cncn1)C C(C(=O)N(C1(C(=O)NC(C)CCCCO)CC1)C)(C(C)C)SC n1(CC(N2CC(CNC(=O)C=CC(F)(F)F)C2)=O)cc(F)ccc1=O c1(NCC#CC)[nH]c(=NCc2c(S(N)(=O)=O)ncn2C)nc2c1ncn2CC C(=O)(C1=CC2(CCN(C(C3(C)CCCN3C)=O)C2)C1)NC1CC2(CC(OC)C2)C1 c1(NCC)ccc(C(=O)NCC(C)NC(c2cccc(OC)c2)=O)cc1[N+](=O)[O-] c1(NC(=O)C(N2CC(Oc3ccccc3)C(C#N)C2)=O)cc(F)ccc1C1CC1 CON(C(=O)C(CNC(C1CCC1C#N)=O)CC1CC1)C(C)C C(=O)(C(C(C)(C)C)NC(N)=O)N1CC(C)CC(NC(C(COC)(F)F)=O)C1 C1(NC(CCC2(C)CN(C(C3(CC=C)CC=CC3)=O)C2)=O)CCN(C)C(C)C1 c1(OCC)ccc2c(n1)NC(C(=O)NCCCCCNC(=O)CCCC(C)C)C2 C1(CCNC(C(CC)CC)=O)CCN(C(c2ccn(CC)n2)=O)C(C)C1 Cc1cccc2ncc(-c3nc(CC(n4ccc(=O)c([N+](=O)[O-])c4)C4CC4)no3)n12 C1(C(=O)NCC(CC)NC(C2CN(S(=O)(=O)C(F)F)C2)=O)CN2CCN1CC2C N1(C(c2cc(Cl)cn2C)C(=O)NCCOC)CCCCC(N2CCCC2)C1 C12(CNC(c3cnn(C)c3F)c3n(CC(=C)C)nnn3)CCC(CC1)C2 N1(C(c2ccc(SC)o2)=O)CCCC(CCNC(=O)Cc2ccsc2)CC1 C(=O)(C(C)CCN(C)C)NC1(CNC(C2(C)CC(=C)C2)=O)CC1 C12(CNC(C3(COCC)CC3)=O)CCC(C(=O)NC(C)C)(CC1)CO2 C(N=c1[nH]cnc2cc(C)[nH]c12)C1(F)CC(NC(C(C2CCOC2)OC)=O)C1 c1(C(=O)NCC2N(C(C(=O)NCC)=O)CCCC2C)c([N+](=O)[O-])cnn1CC C1(C)(CNC(=O)NCCc2ccc(NC(C)=O)cc2)CCC(F)(F)CC1 C1(NC(c2cccn3ccnc23)=O)CN(C(C2C=CCS2)=O)C2CCCC12 C1(CNC(CC2C(C)(C)CCO2)=O)CC12CCN(C(=O)Cn1cc(CO)nn1)C2 C1(CCNC(C2(C(C)=O)CC2)=O)CCN(C(C2(F)CCCC2)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCc1c(C(=O)NCC(CCCCC)(C)C)occ1 C1(NC(C(=O)NC(C)C)=O)CCN(C(=O)CC2COCC2(C)C)CC1F N1(C(CNC(=O)OC(C)(C)C)=O)CC2CCC2(NC(C2(C)CCCS2)=O)C1 N1(C(=O)CSc2nncn2C2CC2)CCCOC(CNC(c2ccncn2)=O)C1 C1(O)(C(C)NC(=O)CCc2cnn[nH]2)CN(C(c2cc(-c3ccccn3)ns2)=O)C1 c1(COC)cccc(C(F)(F)C(=O)NCCC(C)NC(c2ccc(C#N)s2)=O)c1 CC1CC(NC(=O)CC2CCOCC2)CN(C(=O)CCc2cccnc2Cl)C1 C1(CNC(CSC(C)(C)C)=O)CC12CCN(C(=O)Cn1cnc(C#N)n1)CC2 CC(C)C(=O)C(=O)N1CCCCC1CCNC(=O)CC1CC=CCN1C N#CC1CN(C(C2CN(Cc3ccc(F)c(Cl)c3)CCC2O)=O)CCO1 C1(CNC(c2c(C(C)C)n(C)nc2)=O)CN(C(=O)C(C)(Cl)Cl)CCC12CCC2 N1(C(CNC(C(CC)C)=O)=O)CCC2CCCC12C(N1CCC2(CC1)N=N2)=O CC#CCCCC(=O)NCC(C)(C1CC1)NC(=O)CCOc1ccccc1 c1(CSc2ccc(N(CC)CC)cc2)nc(C)c(C(=O)NC2CCOCC2)s1 N1(C(CSCCC(C)C)=O)CC=C(CNC(=O)C(c2cccc(N)c2)C)CC1 CN1CCCC1CCC(=O)NCc1occc1C(N1CCC1C1CCOCC1)=O c1(C(=O)OC)sc2ncnc(NC(C)CN(C(=O)CCn3ccnn3)C)c2c1C C=C(C)CC(C(=O)N1CCOC(CCNC(=O)C(C)CC#N)C1)OC c1(C(N2C(CNC(=O)CCC(N)=O)CC(OC)C2)=O)nsc2ccc(C)cc12 CCC(C)C(CNC(=O)CC(CNC(C1CCC1C(C)(C)C)=O)C1CCC1)OC Cc1cccc2ncnc(N3CCCC(C4CC4NC(C4CC=CCC4)=O)C3)c12 c1(C(=O)NC(C2OCCN(C(c3ccc(C)s3)=O)C2)C)cccc2ncnn12 C(N=c1[nH]cnc(=N)[nH]1)C1CN(C(COC)=O)CC1C.c12ccc(cc1)OC2 N1(C(C(C)OCCCC)=O)CCN(C(C2(SC)CC2)=O)C(CF)C1 Cc1ccc(S(=O)(=O)CNC(c2ccc([Si](C)(C)C)cc2)=O)cc1 C1(NC(C(CN(CC)CC)F)=O)COC2(C1)CN(C(c1cc(C)cc(C)n1)=O)C2 c1(CNC(C2CC(CCC)C2)=O)ncc(C(=O)NCC(c2nncn2C)C)cn1 N1(Cc2cn(C3CCN(C(C(CC)(C)CO)=O)CC3O)nn2)CCc2ccccc21 C1(C(=O)NC2(C(CNC(=O)CC3CC(O)(C(F)(F)F)C3)O)CC2)CC2CCC1C2 N1(C(C=CSC)=O)CCCC(N(C)C(c2cn(Cc3ccccn3)nn2)=O)CC1 C1(C(N(CCCCC)C)=O)(C(=O)OC)CCCN1C(=O)CC1(O)CCCOC1 c1(CNCCC(=O)OC)cc(C)cc(C)n1.C1(C(=O)NC)(OCC#C)CCCCC1 c1(CC(=O)NC2CC(CCNC(C=C(COC)C)=O)C2)nnc(S)n1C Cc1nc(N2CCN(C(c3ccccn3)=O)CC2CCO)c2c(C)csc2n1 C1(C(=O)NC2C3N(C(CC(=O)NC)=O)CC(CC3)C2)CNC(=O)CC12CCC2 C1(CNC(C(CCC)OC)=O)CCCCCN1C(c1ccnc(O)c1)=O c1(NC2CCN(C(C(C)n3cccn3)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 Cc1n[nH]c(=NC(CCN(C)C(c2ncoc2C)=O)C(C)C)o1 C(=O)(CC1=NNC(=O)C1)N1C(C)(C)C(CNC(=O)Cc2cc(C3CC3)on2)CC1 N1(C(COCC=C)=O)CCC2(CC1)CCN(C(=O)C(CC)(CC)CC)CC2 c1(C(=O)NCCN(C(C2CCS(=O)(=O)N2)=O)CC)ccc2c(n1)OCC(=O)N2 C(C#Cc1ccccc1)N1CC(n2cc(CNC(C(CC)OCC)=O)nn2)C1 CC1CCC(CC(N2CC(OCCNC(=O)CC3CSCCO3)C2)=O)O1 Cn1c(=O)n(CCC(=O)NCC2(NC(C3(CCO)CC3)=O)CC2)c2ccccc12 N1(C(CC)C(=O)NC(C)CCNC(=O)Cc2cnn(C)c2)CCN(CCO)CC1 C1(CC(=O)NCC(=O)NCCOC)CCCN(C(c2cc(C(C)C)on2)=O)C1 C12(C(=O)NC3CC(CC(N4C(CC)C(C)CC4)=O)C3)CCC(C1)OC2C N1(C(C(C)N=[N+]=[N-])=O)C2CCC(C2)C1C(N1CCCOC(CO)C1)=O C(CN=c1[nH]nco1)N(C(CC)=O)C(c1[nH]c(O)nc1C)CC1CCCC1 N1(C(C2(C#N)COC2)=O)C2CCC1CC(NC(c1cccnc1OCCO)=O)C2 c1(NCC2CC(C)NC(=O)C2)[nH]c(=NCC2OCCC2(C)C)nc2scnc12 C1(NC(CCCOCC=C)=O)CC(NC(=O)Cn2ncc(Cl)c2C)C12CCC2 CC1OCCCC1C(N1CC(N2CCCC2)C1)=O.C1C(=O)N1 C1(C(=O)NC(CC)CN(C(=O)OC)C2CC2)CCCCN1C(=O)CCC1CCC1 C1(C)(C(N(CCC)CCNC(C2(SC)CCC2)=O)=O)CC(O)CN1C S(=O)(=O)(c1c[nH]ccc1=NCc1cn(C)nc1I)N1CC(C)SCC1 c1(C(N(CC(C)O)CCNC(CN(CCCCCC)C)=O)=O)ccc(CC)nc1 C12(CNC(c3cc(CC(C)C)on3)=O)CCCC1N(C(c1occc1F)=O)CC2 O=C(CCC(CF)CF)N1CC2CCC(C1)N2C(C12CSCC1C2)=O c1(OC)cc(C(=O)N(C)CC2COCCN2C(=O)CC2CCCOC2)ccc1F C12(C(=O)NC(C3CC3C(=O)N(C)C(C3CC3)C3CC3)C)CCCC1C2 CCCCC(O)CCC(=O)NC(C1(O)CCN(C(C2CCCC2(C)C)=O)CC1)C C1(C(=O)NCc2c(C(=O)NCc3nc(C)nn3C)n[nH]c2)CC2(CC(=O)C2)C1 N1(C(c2csc(C(F)F)c2)C(=O)NCCOCC)CC=CCCC(C)(C)C1 c1(NC(c2c(CC)nc[nH]2)=O)ccc(Sc2ccc(Cl)nc2)cc1 C1(C(=O)NC23CC(NC(CN(CC(C)(C)C)C)=O)(C2)C3)CCCCNC1=O N1(C(C2N(C(C)C)C(=O)CC2)=O)CCC(CNC(C2CCC(O)CC2)=O)C(C)C1 N1(C(CN(CC)CC)=O)CC(C(=O)NCC(O)CN(C)C)C(O)C1 C1(C(=O)NC(c2cn(C)nn2)C)CN(C(C2CCCSC2C)=O)CC1C1CC1 c1(CC)nc(N2CC3C(C(=O)NC4CONC4=O)C3C2)c(F)c(Cl)n1 CCCC(C)(O)CC(=O)N(CCC(=O)NCC(C)CC(C)C)CC C(C(C)(C)C(=O)NC1CCC(CCNC(c2oc(CC(C)C)nc2C)=O)C1)SC C1(C(N2CCC(C[SH](C3CCCC3)C)C2)C(=O)NCC)CC2C=CC1CC2.OCC N1(C(CNC(CCC#C)=O)C(F)F)CCN(C(c2cc[nH]n2)=O)CC1 c1(C(=O)NCC(=O)NC2CCCCCC2CO)cccc2cncn12 c1(CC)n[nH]c(C)c1S(=O)(=O)NCC1COCO1 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C(c2ccco2)=O)C(CCO)C1 C1(C(=O)NCC(C)NC(C2(c3ccn(C)n3)CC2)=O)COC2COCC12 CCS(=O)(=O)CC(=O)N1CC2CC2C1C(=O)N(C)Cc1cc(OC)no1 C1(NC(CC(C(C)C)C)=O)C2CCCC1CC(NC(=O)CCc1cnccn1)C2 C12(CNC(C=C(CCC)C)=O)CCCC1CCN2C(c1cc(Cl)cnc1C)=O C1(C2CC2)(CNC(C(C)NS(CCC)(=O)=O)=O)CCN(C(=O)CCC2(C)CC2)C1 c12ocnc1C(=O)NC2.c1ccn(CO)n1.C(C(=O)NC1CCC1)NC(C)=O C(CCCCC(=O)N1CCC(CCC(N2CC3CC2C3)=O)C1)=CC N1(C(C=CC)=O)CC23CCCCC2(C1)CN(C(c1ccc2c(c1)N(C)CC2)=O)C3 c1(CNC2CCC(CC(=O)NC(C#C)C)CC2)cc(F)cc([N+](=O)[O-])c1 c1(COC)nn(C)cc1CNC(c1oc(C)c(C(=O)NCCSC)c1C)=O C(=O)(C1=CCCCO1)NC(C1CC(NC(c2ncc(F)cc2F)=O)C1)C N1(C(C)C)C(=O)CCC1C(=O)CN1CC(C)C1(C)C C1(NC(Cc2cccc(OCC)c2)=O)CC2CC(NC(c3csc(=N)[nH]3)=O)C2C1 c1(CC)cc(C(=O)N(C(C)CCNC(C2(C#N)CC2)=O)C)nn1CCO Cc1cc(C(N2CCC(C)(CNC(C3CC4(CC4)C3)=O)CC2)=O)n2ncnc2n1 N1(C(CC2CCC(=O)C2)=O)CCC2(CC1)CN(C(=O)CC1CC3(CCC3)CO1)C2 N1(C(C2CN(C(c3oc(C)c(CO)c3)=O)CC2(C)C)=O)CC(C)CCC12CC2 c1(C(=O)NC2C(NC(C)=O)CC2)nc(C)ccc1F N1(C(C2(NC(c3cocn3)=O)C(C)(C)C2)=O)CCCNC(=O)C1 CC1CC1N=c1[nH]c(=NCC2(N(C)C)CCOCC2)[nH]c2cccnc12 c1(C(=O)NC2CN(C(c3c(C)noc3)=O)C2)ccc(N2CCNC(=O)C2)c(F)c1 N1(C(C(CF)N(C(C)=O)C)=O)CC2CC1CN2C(=O)COCC(C)(C)C C(=O)(C(CCCC)C(C)C)NCCc1c(CNC(CC(C=C)CC)=O)nco1 c1(C(N2CC(C)OC(CCNC(=O)CCP(C)(C)=O)C2)=O)ccc(N=[N+]=[N-])cc1 c1(C(N(C)CCNC(=O)C(O)CCS(C)=O)=O)n[nH]c2c1CS(=O)(=O)CC2 C(C(C)(C)CCNC(=O)C(C)C(F)F)NC(c1n(C(CC)C)ncc1)=O C1(OCCCCC(C)=O)CN2CCC1(F)CC2 c1(C(C)C)ccc2c(c1)CCCN2C(c1cc(C(F)(F)F)c(Cl)cn1)=O c1(C(N2CC(NC(c3cc(OCC)n[nH]3)=O)C2)=O)cc2ccc(F)cc2[nH]1 C1(NC(C(C)NC(CC)=O)=O)CCCC(NC(=O)Cc2ccc(C(C)=O)s2)C1 N1(CC(=O)NCC(C)C)CCC(C2CCCN(C(C3(O)CCCC3)=O)C2)C1 N1(C(C2N(C(C3C(C)=CCS3)=O)CC(F)C2)=O)CCCCN(C)CC1 c1(C(N2CC(C)(C)C(NC(c3cc(Cl)ns3)=O)CC2)=O)coc2ccc(O)cc12 N1(C(c2c(C)ccc(N)c2)=O)CC2CC(NC(C3C(Cl)(Cl)C34CC4)=O)CC(C2)C1 c1(C(=O)NC2C(CNC(c3c(CC)c[nH]c3)=O)C2)cccn(CC(C)C)c1=O c1(CC)nc(C)n(C)c1C(=O)NCCN(C(c1ccnc(Cl)c1O)=O)CC CC1CCCN1CC(=O)N(CC(F)F)C1CC1 C=C1CC2CC1CN2C(=O)C1=CCN(C(=O)CCNC(=O)COC)C1 N1(CCNC(=O)N(C2N(C(=O)OC(C)(C)C)CC2)C2CC2)CC(=O)NC1=O N1(C(CC(=O)OC)=O)CCC(C(=O)NCC2CC3CCC2CC3)CC1(C)C N1(C(c2c(-c3c(F)ncc(COC)c3)cncc2)=O)CC2CNCC1COC2 c1(OC)cc(C(C)NC(C)C(O)Cc2ccccc2)ccc1OC(F)F c1(C(C)NC(C2(F)CC=CC2)=O)ccc(CNC(=O)CC2CC3CCC2O3)cc1 n1(C(N(CCOC)CCNC(c2cc(=O)cc[nH]2)=O)=O)nc(C)ccc1=O c1(C(=O)NCC(CNC(c2cc(C)n(C(F)F)n2)=O)F)cn2ccnc2s1 C(N=c1[nH]c(=N)[nH]c2[nH]cnc12)C1CCCCC(C(C)(C)C)C1 C(=O)(C(C)C(C)S(C)(=O)=O)N1C2CN(C(c3ccc(OCC)cc3)=O)C(CC2)C1 N1(Cc2cncc(OC)c2)CC2CCN(C(c3cc(Br)ccn3)=O)C2C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CC(C)N(C(C3COCCN3C)=O)C2C1 CCCC(CCCNC(c1cccnc1)=O)NC(c1cccc(O)c1Cl)=O C1(C(=O)NCC2N(C(C3C(C(=O)NCC#C)C3)=O)CC=C2)Cc2cscc2C1 c1(CC(=O)NCC2CNCC2n2ccnc2)cnc(-c2cccs2)s1 N1(C(C(C(C)C)C)=O)CCOCC(F)(CNC(c2ccc3nonc3c2)=O)C1 c1(C(=O)NC(c2ccccc2)CC#C)ccc(Br)cc1C(C)=O Cc1cc(C(=O)NCc2nc(C)c(C(=O)NCCN=[N+]=[N-])o2)c(C)cn1 C1(NC(=O)NCc2ccc(C3C(C)C3)o2)COC2(CCC2)C1O N1(C(c2ccc(P(C)(C)=O)o2)=O)CCC2(CCN(C(=O)C=CC3CCOC3)C2)C1 c12ccccc1NC2=O.C(C(C)C(=O)OCC)N(C(CN(CCC)C)=O)CCC c1(C(N2CCN(Cc3ccc(Br)cc3I)CC2)=O)cccc(Cl)c1Br c1(N(CCOC)CCNC(c2ccc(C(C)(C)C)cc2)=O)ncnc(Cl)c1CO Cc1sc(=O)n(CCC(=O)N(C2CCCN(C(=O)C(C#N)CC3CC3)C2)C)c1C N1(C(c2cnc(C)[nH]2)=O)CC2=C(C1)CN(C(C1CC3(CCC3O)C1)=O)C2 Cc1cc(C(=O)NC2(C)CC(NC(c3c[nH]c(C#N)c3)=O)C2)ccc1Br c1(C(=O)NCCC(C)NC(c2cc(C)cc(C)c2O)=O)cccc(P(C)(C)=O)n1 C=CCC(CC(F)F)C(=O)NC1CCCCC1NC(c1ccncc1F)=O c1(CC(=O)NC2(CNC(c3c(C)[nH]nc3Cl)=O)CCOCC2)nc([N+](=O)[O-])n[nH]1 C1(CNC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)CCCc2cnn[nH]2)CCC1C C1(CC#C)(C(=O)NCc2cccc(NC(C3CCCO3)=O)c2)CCCOC1 C(CCC(C)(C)NC(=O)C=CC(C)(C)C)NC(C1C(C)C1)=O c1(OCC)nc(NC(CNC(=O)C#CC(C)C)C2CCC2)ncc1C N1(C(c2c(C)[nH]cc2)=O)CCOCCC1C(=O)NCCc1ccncn1 c1(NC(C(C2CCCCCC2)N(C(CC)CSCC)C)=O)c(C)cc(C)cc1C CN=C(NCCc1ccccc1[N+](=O)[O-])N1CCC(c2ccccc2)C1 C(C)(CNC(=O)C(CC)OCC)(CC(C)C)NC(c1c(C)nc(CCC)o1)=O Cc1nc(S(=O)(=O)N2CCNC(c3cccs3)C2)ccc1C(=O)O C=CC(C)(C)CCCNC(=O)C(C(C)OC)NC(c1cccc(O)c1)=O c1(CC)[nH]ccc1C(=O)N(CC(=O)NCCn1cc(C)cn1)CCOC CC(C)CCCCC(=O)N1CCCC1CNC(c1ccc2nccn2c1)=O C1(C(N2CCCN(CCNC(CC3CC(SC)C3)=O)CC2)=O)CC2(C1)CC(F)(F)C2 CC1CN(C(=O)CCOCC(F)(F)F)CCC1NC(C1(c2cc[nH]n2)CCC1)=O c1(C(=O)NC2C(O)(C(=O)OC)CCC2)sc2nccc(C)c2c1C N1(C(CNC(C)=O)=O)CC(C)C1C(=O)NCC(c1cscn1)O N1(C(c2c(CNC(C3(OC(C)=O)CC3)=O)cnn2C)=O)CCCN(C)CC1C c1(OC)cc(O)ncc1C(=O)NC1CC12CC(NC(=O)C(C)N(C)C)C2 Cc1scc(C(=O)NC2(CNC(=O)CC3CCC(O)C3)CCOCC2)c1C c1(C(=O)NCC(CNC(c2c(C)onc2)=O)C)[nH]c2c(c1C)CCCC2 C12(CCC1)CC(=O)N2.C(C(=O)N(CCC(C)O)CCO)(C1CC1)SC C1(C)(NC(C(=O)NCCS(=O)(=O)NC(C)C)=O)CC(F)(F)C1 C1(C(C)NC(c2cocn2)=O)CCN(C(=O)CCC2CCCCCC2)CC1 CON1CCC(C(=O)NCC2CC2CNC(C2(c3ccnc(Cl)c3)CC2)=O)CC1 Cc1cc2c(C(=O)NCC3(O)CN(C(c4cnc(C(C)O)s4)=O)C3)cccc2o1 C=CC(CCC)CC(=O)NCCN(C(=O)C(C)CCC)CC O(NC(=O)CC1C(NC(C2(F)CCOC2)=O)CC1O)CC(N)=O N1(C(CN(C(=O)OC)C)=O)CCN(C(C2CCCC(C)(C)C2)=O)C(C(C)(C)C)C1 N1(C(Cc2cc(C)ccc2)=O)CCN(C(=O)COc2ccc(F)cc2Cl)C2CC12 C1(CC(=O)NCC(CNC(c2c(C)csc2Cl)=O)O)CC(C)(C)OC1=O c1(OC)ncc(C(=O)N(C)CC2CCCN2C(c2cc(Br)no2)=O)cn1 CCCCC(C(=O)N1CCN(C(C2CC(COC)C2)=O)CC1C1CC1)NC(N)=O C1(NC(CCc2n(C)cnc2)=O)CCC2CC1CN2C(c1coc(O)n1)=O c1(C(=O)NCCCOCCN(C)C(C2CC2c2cnn(C)c2)=O)cc(O)nc(Cl)c1 N1(C(CC2CCN(C(C=NOC)=O)C2)=O)CCCCCC1.C1(O)CCCC1CF C1(NC(c2cc[n+]([O-])cc2)=O)CCCN(C(=O)CC2CCCN2CCF)CC1 S(=O)(=O)(c1ccc2c(c1)OCCO2)Nc1c(N)cc(Cl)cc1Br N1(C(c2n(CC)cnn2)C(=O)NCCCSC)CCC2CCC(O)C1C2 O=C(N=c1cc(-c2ccccc2OCC2CCOC2)o[nH]1)C#Cc1ccccc1F C(=O)(CC(C)(C)CN(C)C)NC1C(C)CN(C(=O)C(CO)N(C)C)C1 c12ccnc(n1)CC(C)N(C)CC2=O.C1(CC(=O)OC)CC(C)=NO1 c1(C(=O)NC(CN(C(C(C)OCCOCC)=O)C)CC)cc(O)cc(N)c1C CC(CC(=O)NCCN(C(c1cc(O)ccc1C(N)=O)=O)C1CC1)C(F)(F)F CCCCC(C(=O)NCCSC)NC(c1ccc(C)c(O)c1)=O c1(C(N2CC(NC(C3CCCC(C)CC3)=O)C2)=O)nnc2ccccc2c1N c1(OC)c(Cl)cc(C(N2CC(NC(C3CC(N(C)C)C3)=O)C2)=O)cc1Cl c1(C(C)SCC)cn(Cc2c(CC(=O)NCc3ccccc3)nco2)nn1 c1(C(=O)NCCCNC(C2C(c3cn(C)nn3)C2)=O)coc2c1CCCC2 c1(C(=O)NC2(C)CN(C(C3(OC)CCOCC3)=O)C2)cnn2ccc(Cl)c(F)c12 C1(CC(=O)NCC(CC)CO)CCCN(C(C2CCC(C)O2)=O)C1 C12(NC(c3cc(Cl)c[nH]3)=O)CCC(CC1n1cc(CN3CCCSCC3)nn1)C2 C(=O)(CC(C)CC(=O)NC(CC1CC1)C(=O)NCCCC1(O)CC1)OC C1(NC(COCCC)=O)CCC(NC(=O)C=CC(c2ccccc2)=O)CC1 C1(CC)CC(O)CCN1C(=O)C(C)NC(=O)C(C1CC1)SC c1(C(N2C(CNC(c3ncc(NC)nc3)=O)COCC2)=O)ccn2ccnc2c1 C1(C(=O)NCc2c(CCNC(c3cc(C)no3)=O)ocn2)CN(C)CC(C)O1 c1(OC)cc(C(=O)NC2CC2CNC(C2(C)CC2)=O)ccc1C(F)F N1(C(C(C)NC(=O)NC)=O)C2CCC1CC(NC(C1(C(C)(F)F)CC1)=O)C2 CN=C(NCCOC(C)=O)N1CCC(Cc2ncccn2)C1 C1(NC(c2ccc(NCc3sccc3Cl)nc2)=O)CNC(=O)C12CC2 C1(NC(c2cn(C(C)C)nc2)=O)CC2C(NC(c3ncc(C(F)F)s3)=O)C2C1 O=C1CCN(CC(N2CC(CO)(NC(C3CCCC(F)C3)=O)C2)=O)C(=O)N1 c1(NCc2cccc(C(=O)OC)c2)ncc(Cl)nc1Cl.C1(=O)CO1 C1(COC)CN(C(c2ncc(N)cc2C)=O)CCN1C(c1cc(C)cs1)=O c1(C(=O)NC2CCN(C(COCC=C)=O)C(C)C2)cnn2cccc(Cl)c12 N1(C(c2c(OC)ccc(OC)c2)=O)CC2CCCN(C(=O)CC3C=CCC3)C2C1 N1(C(c2cccc(C)c2C)=O)CCC2(CC1)CC(N1CCC(C#N)C1)CO2 C(=O)(CC(C)(C)C)NC1CC(OCC(=O)Nc2ccc(COC)o2)C1 N1(C(Cc2cnc(C)[nH]2)=O)CCCN(C(=O)C(CC(C)C)NC(N)=O)C(C)C1 C#Cc1cc(NCCC2CN(C(=O)CN=[N+]=[N-])CCO2)ccc1Cl C=C(C)C(CC(=O)NC(CNC(=O)Cc1ccnn1C)C(C)C)OCC N1(C(C2CC(C)OCC2)=O)CCOC2(C1)CN(C(C1(CO)CC1)=O)C2 N1(C(COCC=C)=O)CCC(C)(C)C1CC(N1CC(C)(C)C1COC)=O c1(C(=O)NC2CC(F)(CNC(C(C(C)C)SC)=O)C2)cc2ncccn2n1 n1(CC2(CCCc3noc(C)n3)CC2)ccc(C(=O)NC(C2(CC)COC2)=O)c1 Cc1cnc(C(=O)NC2CCN(C(c3cnn4cc[nH]c34)=O)C2C)c(C)c1 CC1CC(NC(c2cc(C(F)F)on2)=O)CCN1C(=O)COC(F)(F)C(F)(F)F C1(CC(C)C)(CNC(=O)Nc2ccccc2Nc2ccccc2)CCCOC1 n1(CC(=O)NC2C(NC(c3ccc(CC)s3)=O)CC2)nc(C)ccc1=O N1(C(CC(C)c2ccco2)=O)CCCCC(N(C)C(c2ccc(F)o2)=O)C1 CCC(CC(=O)N(CCC(=O)N1CCc2ncccc21)OC)C(F)F Cc1c(N2CCN(C3CCCCCCC3)CC2)ncnc1Cl C1(C(C)C)CN(C(C2(Cl)CC2)=O)CCN1C(c1cc(C(N)=O)cs1)=O N1(C(C(c2ccnn2C)C)=O)CCN(C(c2c[nH]nc2C)=O)C2(CC2)C1 C1(NC(c2cnn[nH]2)=O)CCCCCC1NC(=O)C(c1ccccc1)O c1(C(=O)NC(C(C)NC(c2c(Cl)cc(C)s2)=O)(C)C)ccc(OCCF)cc1F c1(C(C)C(=O)NC2C(C(=O)NCCC(=O)NC3CCC3)C2)ccc(F)c(Cl)c1F CC#CCCCC(=O)NC(C1CN(C(=O)C2=NNC(C(F)(F)F)C2)C1)C CCCC(C(=O)NC1(c2nnnn2CCCF)CC(CO)C1)NC(=O)OCC CC1CN(C(C2CCC(C(F)(F)F)CC2)=O)CCCN1C(=O)C1=CSCCO1 c1(C(=O)NC2CCC(NC(C(C3CCC3)OCC)=O)C2)c(OC)cccc1C N1(C(c2cc(C)sc2)=O)CCN(C2CCCN(C(c3cccn3C)=O)C2)CC1 c1(OC)cc(C(N2CCC(C(C)NC(=O)COc3ccon3)C2)=O)cc(C)n1 C(CN=c1[nH]nc(C2CC2)o1)C1CC(C)N(C(c2cn3ccccc3n2)=O)C1 Cc1cccc2cc(C(=O)N(C3CN(C(c4ccncn4)=O)CC34CC4)C)oc12 C1(CC)CN(C(=O)CCc2ccc(Cl)s2)CCC1NC(c1coc(C(N)=O)c1)=O N1(C(CC=C)=O)CC2CC1CCN2C(c1ccc(NC(=O)C(C)(C)C)nc1)=O c1(NCC=CCOCC)cc(N2CCN(CCO)CC2)nc(C(F)(F)F)n1 C(=O)(C1=CC2(CCOC2)C1)NCCNC(CCCC1C(C)C1)=O C1(C2=CCCC2)CC(=O)N1.C1(COC)COCCN1C(=O)Cc1cnoc1 CCC(C(=O)N1CCC(CNC(=O)CCCc2nc(C)cs2)C1(C)C)C(C)(F)F C(c1cc(F)cc(F)c1)=CC(=O)NCCN(C(C1CCCCC1F)=O)C1CC1 N1(C(C2C(C(C)C)C2)=O)CC(=O)NCC1C(=O)NCCc1nc[nH]n1 c1(C(=O)NCc2occ(C(N(c3ccccc3)CC=CC)=O)n2)cnccc1C#N C1(O)(C(C)CNC(C23CC(C)(C2)C3)=O)CCN(C(=O)CC2(C)CC2)CC1 S(=O)(=O)(CC(=O)NCC1CCCC1NC(=O)C(=Cc1ccco1)C)N(CC)CC C1(C)(CNC(C2OCCC(N(C)C)C2)=O)CCN(C(C2(Cl)CC2(F)F)=O)CC1 N1(C(c2ccccc2)=O)CCN(C(C2CC2(Cl)Cl)=O)CC1CC(F)(F)F.CCO c1(C(N(C(C(=O)N(CC(=O)OCCC)C)C)CC)=O)cc(CC)[nH]n1 c1(C(=O)NCC2CN(C(C(F)=C(C)C)=O)C(C)C2)cccn2nnnc12 Cc1ccc2scc(C(N3CCN(C(=O)C4=CCCC4)CC3CF)=O)c2c1 C(=O)(C1=CCCCCC1)N1CCC(C(C)NC(C2CC(C)SCC2)=O)C1 N#Cc1c[nH]c(=NC2CN(C(C3COCCO3)=O)CC23CCC3)c2sccc12 C1(C(=O)OC(C)(C)C)CN(CC2C(C)CCNC2=O)Cc2ccnn2C1 C1(CCC(=O)OC)COCCN1C(=O)N(C1(c2cc(C)[nH]n2)CC1)C C1(C(C)NC(=O)C(O)C2CCC2)CCN(C(=O)C=CI)C1 C1(NC(C(C(C)C)(C)C)=O)CN(C(C2C=CC=CC=C2)=O)C2(CCOCC2)C1 C1(NC(C(C)Sc2ccccn2)=O)CCC(CNC(=O)C(O)c2ccco2)CC1 CC1(C)CCCC1C(=O)NCC(O)CNC(=O)CCCOc1ccc(F)cc1 C12(C(=O)NC(CNC(C3CC3C(F)(F)F)=O)C3CC3)CCC1CC2 c1(C(=O)NC2CCN(C(C3(F)CCS(=O)(=O)C3)=O)C2)csc2cncn12 c1(-c2cc(C(=O)NCc3nccc(OC)c3)n[nH]2)ccc(F)cc1CO N1(C(c2cc(C)c(C)o2)=O)CC2(CCC(CNC(C3Cc4nccn4C3)=O)O2)C1 C1(C(=O)NC2C3CN(C(c4n(CCC)nc(C)c4)=O)CC32)CNC(=O)CC1C C12(CC(=O)N(CCCN(C(C=CC)=O)CCc3ccccc3)CC)COCC(C1)C2 c1(C(N2CCC(C)N(C(C3CCSC3)=O)CC2)=O)ccc2c(c1)OC(F)(F)O2 N1(C(CCN(C(C2CCC(O)C2)=O)CC)=O)CC2CC1(CO)C2 C(C1COC(C)(C)O1)=CC(=O)NC1(CNC(C2CCC(C)O2)=O)CCOCC1 c1(C(N2CC3C(CNC(=O)C(Cl)=CCl)(C3)C2)=O)ccc(=O)n(CCO)c1 c1(C(c2nnnn2CC(F)F)NCc2nc(C)oc2)ccccc1N(C)C N1(C(C(CC2CCCC2)NC(c2cccc(O)c2)=O)=O)CC2CCC1C(O)C2O c1(C2C(C(N3CCC(C(=O)N(C4(CC)CCCC4)C)C3)=O)C2)ccc(F)c(Cl)c1 NC(=O)CC(C(=O)NCCCC1(O)CCC1)NC(c1n[nH]c(O)n1)=O CCCCCCC(COCCOC)(c1nnnn1C1COC1)NCC(C)(C)C c1(-c2cncc(C3CC(NCCN4C(O)CCC4)C3)c2)ccc(Cl)nc1 C1(C)(CNC(C(CNC(c2c(CC)noc2)=O)C)=O)CCC(=O)N1C C1(C)(C(=O)NCC(c2cccc(Cl)c2)NC(C(C)(C)OC)=O)CCCOC1 C(=O)(C1CCOc2c(F)cccc21)NC(CNC(CCC(=C)Cl)=O)(C)C Cn1nc(C2CCC2)cc1C(N1CC2CC2(NC(=O)C=Cc2ncc[nH]2)C1)=O C12(C(=O)NCCNC(c3ccc(OCC(C)C)cc3)=O)CCCN1CC(O)C2 CC(O)(C(=O)NCC1CC2CC1CN2C(C1CC1C1CCC1)=O)C(F)(F)F C(C(C)(C)C#CC(=O)N(C(C)C(C)C)C)NC(COC)=O N1(C(CC2CC(C)C2)=O)CCC(NC(=O)C=CC(=O)NC2CC2)C1(C)C n12nccc1C2C.c1(C(C2CC2)NC(C2CC2)C2CC2)nnnn1C1CC1 N1(C(C2(COC)CCCO2)=O)CC(NC(C2SCCS2)=O)C2(CCOCC2)C1 c1(C(=O)NC(CCNC(c2c(C)n(C)nc2)=O)C)nccc2ccsc12 C1(CNC(c2cn[nH]c2)=O)C(C2CC2)CCN1C(=O)CN1CCC(F)(F)C1 N1(C(Cc2ncc(C)o2)=O)CCC(NC(=O)C=Cc2ccc(Cl)s2)C(F)C1 CC(CC(C)(C)C)C(=O)N1CCN(C(=O)Cc2csc(C3CC3)n2)C(CO)C1 c1(C(N(C(CNC(CN(CCCCCC)C)=O)C)CC)=O)c(C)cnn1C(C)C c1(N2C(CCCNC(C3CCCCO3)=O)CCC2)ccc([N+](=O)[O-])cc1Cl CCCC(O)C(=O)NCCCC1CN(C(c2cc(N(C)CC)ccn2)=O)CCO1 Cc1nc2nccc(NCC3(C)CCN(C(=O)Cc4nc(C)c(C)s4)C3)n2n1 c1(CC(N2CC(NC(c3ccc(CC)cc3)=O)C(C)C2)=O)ccc(C)cc1F C1(NC(=O)NCCC(=O)C2CCCC2)CCCC1n1ccnc1 C1(SCC)C(NC(C2CC=CC(O)C2)=O)CCCN1C(=O)CC1CCSC1 C(CCCCC(=O)N(C1CCCCN(C(=O)C(F)(F)C2CCOCC2)C1)C)=CC N1(C(Cn2c(C)ncc2)=O)CC2(COC(CNC(=O)C(c3ccnn3C)C)C2)C1 n1(CC(=O)NCCC(P(C)(C)=O)N(C)C)ccc2ccccc2c1=O N1(C(Cc2cc(C)no2)=O)CCCC2CN(C(=O)CCc3csc(=N)[nH]3)CC12 c1(OC)c(Cl)cc([N+](=O)[O-])c(Cl)c1C(N1CC(N2CCN(C(=O)CO)CC2)C1)=O N1(C(C(CC=C)C)=O)CCc2ccccc2C(NC(C2COCCN2C=O)=O)C1 c1(C(C(=O)NC)N(C2(C#N)CC2)C)ccc2c(c1Cl)OCO2 Cc1cnc(C(=O)NC2(CNC(=O)C3=CCCCO3)CCCCC2)cc1C#N C1(NC(c2cccc(CC)c2C)=O)CC(C2CCN(C(c3cccn3C)=O)C2)C1 Cc1ncc(CN2CCC(c3ncon3)CC2)n1-c1ccccc1 c1(N(C(=O)CCCN2CCC3CC3CC2)C(CC)=O)ccc(C(F)(F)F)c(F)c1 c1(C(=O)OC)nc(Br)ccc1NC(C1(C)CCN(C(c2cccc(F)c2)=O)C1)=O c1(C(N(C(C(c2cccc(C(F)(F)F)c2)C)=O)C)=O)ccc(C(=O)CF)cc1 c1(C(N2CC(CN(C(C3C(C)OCC3)=O)C)C2)=O)cc(F)cc([N+](=O)[O-])c1 CN1CC=C(C(=O)NCCCNC(c2conc2C(C)(C)C)=O)C1 C1(CNC(c2cc(Cl)no2)=O)CCCC(CO)C1.C12CC(C1)C(=O)NC2=O.C1(N)CC1 C1(NC(C(CCOC)OC)=O)CN(Cc2cccc(C)c2)CC1(F)CN(C)C C(=O)(C1=C(C)OCCS1)NCC1CCCC(C(=O)NCC2(OCC)CCC2)C1 N1(CC(=O)NCC2CN(C(c3ccc(O)nc3)=O)CC2O)CCC(=O)NC1=O C=CCC(F)(F)C(=O)NC1CCCC1CNC(C1C=CCS1)=O CC1CCC(C(N2CC(F)(F)C2C2CC2)=O)N1C(C1C2CCC(F)C12)=O C1(CNC(c2cncc(OC)n2)=O)CN(C(=O)CCCCO)CCN1C C(C(COC(=O)Cc1cn(C)nc1C(F)(F)F)C(F)(F)F)NC(C)=O Cc1nc(C)c(CNC(C2CC(C)N2C(c2cc[nH]c2)=O)=O)s1 c1(C(=O)NC2CC(C)N(C(=O)C=Cc3cncc(O)c3)C2)cccn2ncnc12 N1(C(c2cnc(C)nc2C)=O)CCC2(CC(C(N3CCOCC3C(C)O)=O)C2)C1 c1(CN2CC(F)CC(C(=O)N(CCO)C3CC3)C2)cc(F)cc(Br)c1F C(=O)(C#CC1CCCO1)NCC1(O)CCN(C(Cc2ccc(OC)c(F)c2)=O)C1 N1(C(C=Cc2c(C)cccc2)=O)CCCC12CCN(C(c1nncs1)=O)C2 c1(NC(C2COCCN2CC2CCCCO2)=O)ccc(O)cc1F C12(C(N(C3CCN(C(CC(C)n4ccnc4)=O)CC3)C(N)=O)=O)CCCC1C2(F)F N1(C(C2N(C(C(=Cc3ccncc3)C)=O)CC=C2)=O)CC2CCC2(C)C1 N1(C(C(C)NC(C)=O)=O)CC(N(C)C(c2cnc(-c3cnn(C)c3)s2)=O)C(O)C1 C(=O)(C#CC1(C)COC1)N1CC(C)C(CNC(=O)CN(C)C2CC2)CC1 Cc1cc(C(=O)NCC(C)(C)NC(=O)CC(C)(C)c2ccc(F)cc2)nc(C)c1 CC1CN(C(=O)CCC2CCCN2C)CC1(C)C(=O)Nc1ccc(F)c(O)c1 C1(CN(C(c2cnccc2OC)=O)CC)CCCN(C(C2CC2[N+](=O)[O-])=O)C1 CC12CCOC(CC(N3CC(C)(C(=O)NC(C(O)CO)C4CC4)C3)=O)(C1)C2 N1(C(C=C(CC)CC)=O)CCC2C(NC(c3cc(OC(C)C)ccn3)=O)C2CC1 C1(NC(c2ncn(C)n2)=O)CCCC(NC(=O)C(F)=CC2CC2)C1 C1(NC(Cc2c(OC(C)C)cccc2)=O)CN(C(C2CC2F)=O)C2CCCCC12 N1(CCOC)CCN(C(c2cc(Br)ncc2F)C(=O)NCC2CCOC2)CC1C CCC(C)CN=C(NC1CCCCC1)N(C)CC1(C)CCCCC1 Cc1ccc2c(c1)C=C(C(=O)N1CC(NC(C3CN(C)CCO3)=O)C(C)C1)CO2 Cc1nc2c(C(=O)N(CCNC(=O)C(C)CC3CCCO3)C3CC3)cccc2o1 CCCC(CNC(C1C2COCC12)=O)NC(=O)C=C1CCSCC1 c1(C(N2CCN(S(C3(CC=C)CC3)(=O)=O)CC2CC)=O)c(Br)cc(Cl)nc1Cl N#Cc1cc(C(=O)NCC23CC2CN(C(c2ccc(CO)o2)=O)C3)c(F)cc1F C1(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CN(C(=O)C(F)(F)CO)CC1O CCCCC(=O)N1CC(C(=O)NC(C(F)(F)F)C2CC2)(SC)C1 CC1(C(=O)NC(C2CCCC2)CNC(c2ccnc(S)c2)=O)CC(C2CC2)=NO1 c1(C(=O)NCC(CC)NC(=O)Cn2cc(Cl)cn2)cc2ccc(F)cc2nc1C C=CCCC(C)(C)C(=O)NCC1CC2CCC1N2C(c1ccc(CC)cc1F)=O c1(C(=O)NC(c2ccc(C)c([N+](=O)[O-])c2)C)cc2c(nc1N)CCCC2 C1(C)(CC)CC(NC(c2n[nH]c3c2CCC3)=O)CN1C(=O)C(C)=C(C)C C1(NC(N(C)Cc2n(CCC)cnc2)=O)CCN(CCOC)CC1 Cc1ccc(C(C)C(N2CCC(CN(C)C(C3CCOC(=O)N3)=O)CC2)=O)cc1 C(=O)(C(CO)C(C)(C)C)N1CC(CC(=O)N(C(=O)OC)CCO)CC1(C)C C1(C(=O)NC(CO)C2CC2)C2CN(Cc3ccc(N4CCCC4)o3)CC12 C1(CNC(=O)NC2(C(c3ccccc3)O)CCOCC2)CC2(C1)CC2(F)F C1(C(N(C)Cc2c(C)n[nH]c2)=O)CCC(C2CC2)N1C(=O)CC1CC(C2CC2)C1 Cc1cc(NC(=O)Cc2cnn(CCNC(=O)OC(C)(C)C)c2)c(O)c(C)c1 C1(C(=O)NC2CC(F)(C(=O)NC(c3cccs3)CC)C2)CCC(C)=C(C)C1 C(=O)(C(C)(C)C(F)(F)F)N1CC(NC(C2(N(C)C)CCCC2)=O)C(CO)C1 CC1=NOC(CC(N2CC(C)(NC(c3cc(CC4CCCCC4)c[nH]3)=O)C2)=O)C1 C#Cc1cccc(C(=O)NCC2(F)CCN(C(=O)C(C)C(F)(F)F)C2)c1 c1(C(N2CC(C)C(NC(=O)Cc3cccnc3)C2)=O)ccnc2c(F)cccc12 c1(CNC(=O)CCCNC(=O)CC2CCOC2)c[nH]ccc1=O N1(C(C2C(CC)OCC2)=O)CC2CC2(NC(c2nccc(C)n2)=O)C1 N1(C(c2nnc(C)s2)=O)CCN(C(c2ccc(Cl)c(F)c2)=O)CC1C1CCCC1 S1(=O)(=O)C2=C(Br)C=CC(=NCC(C)(C)C3CCCC3N1)N2.CN1CCC(CO)C1 C1(NC(COCc2ccc(C)cc2)=O)COC2(C1)CN(c1cc(C)ncn1)C2 c1(C(=O)OCc2nc(N3CCCC3)n[nH]2)cc(N2CCNC2=O)ccn1 Cc1cc(=NC(=O)C2CC(NC(c3cc(O)ccc3F)=O)CCO2)[nH]n1CCO c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC2N=[N+]=[N-])n[nH]c2ccc(Cl)cc12 C1(NC(C(CC)CO)=O)CCCCC12CCCN(C(C1CC(=O)N(C)C1)=O)C2 C1(C)(C(N(C)CC2CCCN(C(C34CC(O)C3C4)=O)C2)=O)CCN(C)CC1 c1(OC)c(Br)ccc(C(N2CC(CC(N3CCC(F)C3)=O)C2)=O)c1F c1(C(N2CC(CC)N(C(c3cc(C)on3)=O)CC2)=O)cc(F)cc(S(N)(=O)=O)c1 Cc1ccc(Cl)c(C(=O)NCCC2CC(NC(c3cccc(Cl)c3N)=O)C2)c1 c1(NC(C2(F)CCN(C(C3(CC=C)CCC3)=O)CC2)=O)ccc2nccn2c1 CC1CC(C)OC1C(N1CCCCC1C1CCCN(C2CCN(C)C2=O)C1)=O c1(C(N2CCC(N3CCCC3)C2)C(=O)NCCC2(C)CC2)cnc(Br)s1.C(CO)N N1(C(c2ccc(C)o2)=O)CCC(C(=O)Nc2cnc(F)c(C)c2)C12CC2 C1(NC(c2cnc3ccsc3c2)=O)CC2CC(C1)N(C(C1(F)CCOCC1)=O)C2 c1(C(N2CCC(C)(C(=O)Nc3cncnc3)C2)=O)ccnc(Br)c1Cl C1(NC(CCC#C)=O)CCC(C(=O)Nc2ccc(OC)nc2)CC1 C1(NC(C2CCN2C2CCCC2)=O)CCN(C(c2cn(C3CC3)nn2)=O)CC1F N1(C(C=CCN(C(=O)Cc2cncn2C)C)=O)CCN(C)C2CC12 c1(C(=O)NCCCCCN(C)C(C2C3CS(=O)(=O)CC23)=O)ccc(F)c(O)c1F CC(CC(C)(C)CO)NC(C1(CF)CCN(C(=O)C(C2CCOCC2)=O)C1)=O C12(CNC(C(CC)OCC)=O)CCC(C1)N(C(=O)Cc1ccc(C)s1)C2 CC1CN(C(=O)C(C)(C)C(C)c2ccccc2)CCCN1C(=O)C(F)F C(CC(N)=O)(C(=O)NCC1(C)CCCCO1)NC(c1cc(CC)nn1C)=O c1(C(=O)NCc2ccccn2)csc2c1CCN(C(c1cccn1C1CC1)=O)C2 C12(CCCOC1)c1cn(nn1)C1C(C=CCC1)C(=O)N2.CCCOCCO Cc1ncc(CCC(N2CC3(CC3)CC2CNC(c2nccs2)=O)=O)c(O)n1 N1(C(C2(SC)CCC2)=O)CC2(C=C(C(=O)NCC3(C)CCCOC3)CO2)C1 c1(CC)ncncc1C(=O)NCC1(F)CCC(NC(=O)C(C)(CO)OC)C1 C(=O)(CCCC(=O)N1CCC(N(C(=O)CC(C)OC)CC)C1)NCCC n1(C(C)C)ccc2cc(C(=O)NC(C)CN(C(=O)CSC(F)F)C)ccc12 C#CCCC(O)C(=O)NC(C)(CNC(=O)CCc1ccc(C)c(Cl)c1)CC(C)C N(C)(S(=O)(=O)N(C)C)CC(=O)NCC1N(C(CC=CC=C)=O)CC(O)C1 c1(SCC)cc(Cl)ccc1CN1CC(NC(c2oc(C3CCC3=O)nc2C)=O)C1 C1(NC(CN(C)C)=O)CC(=O)N(C2CN(C(=O)CCc3cccnc3F)C2)C1 N1(C(CN2CC(C)(OC)C2)=O)CCC2CCCC12C(=O)NC1CCSC1 N1(C(C2(CC(C)C)CC2)=O)CC(NC(c2ccn(-c3cccnc3)n2)=O)C(O)C1 Cn1cc(C(=O)NC2CC2NC(c2cnc[nH]2)=O)c(-c2cccc(F)c2)n1 c1(C(=O)NC(CC)CNC(=O)CC2CC(C)=NO2)nn(-c2ccccc2)cc1C C1(C(N(CCC)CCNC(=O)Cc2c(F)cccc2Cl)=O)CCN2CCCC2C1 N1(C(C=CCC)=O)CCC2(COC(CNC(c3cc4cnn(C)c4s3)=O)C2)C1 c1(C(=O)NCC(n2cc(C3(Cl)CC34CCC4)nn2)C)cccc2c[nH]nc12 N1(C(COC(C)C)=O)CCCC(CO)(NC(=O)C(c2ccc(Cl)cc2)=O)C1 CCC(C)(C(=O)NCC(C1CC1)N(C(=O)Cc1ccc[n+]([O-])c1)C)OC c1(C(C(=O)OCC)(C)C)cccc(C2(NC3CCOC(C(C)C)C3)CC2)c1 CCCC(CCC)C(=O)N(CC(=O)OC(=O)CCBr)C1CC1 Cc1ccc(NC(C)CNC(=O)C(C)NC(=O)CN(C)C(N)=O)cc1 c1(CC(=O)NCCNC(C2C(C)C2)=O)ccc2sccc2c1 C(CC(CC)C(=O)N(C)CC1CN(C(c2ccc(C(C)C)cc2)=O)CCO1)=CC C=CCC(C)(C(=O)NC1(C)CCCN(C(C2CCS(=O)(=O)N2)=O)C1)N(C)C C=CCC(CC(C)C)C(=O)NCC(C)(O)CNC(=O)CC1=CCOCC1 N1(C(C(=O)NCCC2CC2)c2ccco2)CCC(C2CCC2)C1 C(CC(CC)C(=O)NCCC1CCCN(C(c2cc(CC)[nH]n2)=O)C1)=CC Cn1nnc(CNC(=O)C(F)F)c1C(=O)NC1CC(n2cccn2)C1 C#Cc1cccc(C(=O)NC2CC(N(C(=O)CC3CCCCO3)C)C2)c1 C12(CNC(C3C(C)CC3)=O)CCC(C(=O)O)(CC1)CO2 CC(CCC(=O)NC1CCCC(NC(=O)COC2CC2)C1)OC(C)(C)C N1(C(Cn2c(C)cc(C)n2)=O)CCN(C(C2CC(C3CCC3)C2)=O)C2COCC12 C1(F)(C(N(CCCNC(=O)C(F)CC2CCC2)CC)=O)CCN(C)CC1 c1(OCC(=O)NCC(C(C)C)NC(C(Cn2ccc(C)n2)C)=O)cncc(Cl)n1 c1(NC(=O)NC2CCCN(c3ncc(OC(F)F)cn3)C2)c(F)ccc(F)c1F C(C(F)(F)C(=O)NCC(C1CCCCC1)NC(c1cc(C(C)=O)on1)=O)OC c1(C(c2nnnn2C2CCCC2)NCc2ncn(CC)c2)ncc(OC)cc1F c1(N2C(C(C)O)CCC2)ccc2cc(S(=O)(=O)NC3C=CCCCC3)ccc2n1 C1(CNC(c2cccnc2Cl)=O)CCN(C(c2cc(Cl)ncn2)=O)CC1O Cc1ccc(OCCOC(=O)C=Cc2ccncc2)cc1Br N1(C(CC(C)NC(c2ccccc2)=O)=O)CC2(CCN(C(=O)C(C)(C)F)C2)C1 C1(CNC(c2cncc(C)n2)=O)CC(C)(C)CN1C(=O)C(O)C(C)C c1(C(=O)NC2CCCN(c3ncc(C(F)F)cn3)CC2)ccc(F)c(F)c1F C1(C(=O)NCC2C(NC(CCNS(CC)(=O)=O)=O)C2)CC(S(N)(=O)=O)C1 c1(C(=O)OC)c(NCC(C)Nc2ncc(C)c(SC)n2)ncc(C)c1C C1(NC(Cc2nc(C(C)OC)sc2)=O)CC2CN(c3cc(C)[nH]n3)CC2C1 N1(C(CC2OCCN(C(C3(CC(C)C)CC3)=O)C2)=O)CC2CCCCC2C1C C=CCC(C(=O)NCCC1=CCN(C(c2ccc(Br)c(C)c2)=O)CC1)C(C)C C#Cc1c[nH]nc1C(N1CCC(n2cc(-c3ccccc3COC)nn2)C1)=O C1(NC(C=CCOCCOC)=O)CCC2CN(C(C3CC(=O)NC(=O)N3)=O)CC12 CC1CC(CCNC(c2ccc(Cl)o2)=O)CCN1C(=O)COc1cnn(C)c1 NS(=O)(=O)N1CC(C(=O)NCCC(O)CNC(C2CCCS2)=O)C1 C#CCCCCN=C(NCS(C)(=O)=O)NC1CCS(=O)(=O)C1 N1(C(C=CC=CCC)=O)CCCC2(CNC(c3cn(C)c(C)n3)=O)CCCC12 Cc1nc2ccc(S(=O)(=O)N3CCC4(CCC(O)C4)C3)cc2[nH]1 N1(C(C2C(OCC)C2C)=O)CCCC(C(C)NC(=O)C(F)C2CCOC2)C1 C(=O)(C(O)CC1CCCCC1)NC1C(C(=O)OC)(Sc2ccccc2)C(C(=O)O)C1 C1(NC(CCC2CCN(C(C=CC(=O)OCC)=O)C2)=O)CCCCC12CCC2 c1(C(=O)NC(CC(=O)NCC(N(OC)C)=O)C)cc(O)ncc1F c1(CC(N2CCC(NC(CCCCC)=O)(COC)C2)=O)cc(C)ccc1C C1(CNC(=O)C(F)CC2CC2)CC2CCC(C1)N2C(=O)Cc1ccc(O)nc1 N1(C(C(CN(C)C)NC(CCc2ccc(C)o2)=O)=O)CCc2nocc2C1 C12(NC(=O)Cc3cscn3)CCCC1CN(C(c1ncsc1C(F)(F)F)=O)C2 C12(NC(C(N3CCSCC3)C)=O)CCOC(CNC(=O)C3=NNC(=O)C3)(C1)C2 C(=O)(CC(C(C)(C)C)NC(=O)CCC(C)(C)C#N)NCCCC(C)(F)F C1(C(=O)NCC=CC)CN(c2ncc(F)cn2)CCC1O N1(C(CCSCCC)=O)CC(NC(=O)CSCC(C)C)CCC1C N1(c2cccc(C)c2)N=C(C(=O)NCCNC(=O)C(=O)N=S(C)(C)=O)CCC1=O C1(C(N(C2CCN(C)C2)C)=O)CCN(C(c2ccsc2Cl)=O)C(C)(C)C1 C1(NC(C=CCOCCOC)=O)CC2CN(C(=O)C=CC=C(Cl)Cl)CC12 CCCCC(O)CC(=O)N1CCC2(CC1)CC2C(=O)NC(c1ccsc1)(C)C C1(CCNC(c2cccs2)=O)(NC(C2CN(S(CC)(=O)=O)C2)=O)CCCC1 c1(C(N2CC(CC(C)NC(CN(CC)CC)=O)C2)=O)cnc(C)nc1C C=CCCCCC(C(=O)NCCCF)N1CCCCC(Cn2cncn2)C1 C1(C(=O)NCCC=CC=C)CC2(CCN(C(=O)CCC=C(C)C)C2)C1 CC1(C(=O)NCCC2CCC(NC(c3ccc(F)s3)=O)C2)Cc2ccccc2N1 c1(C(=O)NC(C2CCN(C(c3cccc(SC)c3)=O)C2)C)cccc(F)c1O c1(C(=O)NC2CN(C(C3N(CC)CCC3)=O)C(C)C2)cccc(C)c1F C(CCCS(C)=O)NC(CN(C(c1cc(OCC)no1)=O)CC)=O C(=O)(C(CC(C)C)NC(C1(C)CCN(C(C2CN(C(C)=O)CCC2C)=O)C1)=O)OC N1(C(c2ncc(CC)cn2)=O)CC(CN(C)C(c2ccccn2)=O)C2(CC2)C1 C1(Nc2ccc(F)c(Cl)c2F)CC12CCc1cc(Br)ccc12 C1(CC(=O)NCC2CC(F)C2)CN(C(c2ccncc2Cl)=O)CCO1 c1(C(N(CCC(C)NC(=O)CCc2ncc[nH]2)C)=O)ccc2c(c1)C=CS2(=O)=O c1(C(=O)NCCCN(C(c2cc(Br)c(C)cn2)=O)CC)c(C)ccc(C)c1O C1(N(C(=O)CC2OCCO2)C)CCCN(C(C2(C3CCC3)CC2)=O)CC1 CC1(C)CC(=O)N(CC(=O)NCCCOCCCNC(C2CC2(Cl)Cl)=O)C1=O C(=O)(C(CC)C(=O)NC(c1ccccc1)C(=O)NC1(CO)CC2(CCC2)C1)OCC C1(CC)CCCC1(C)C(N1CCC1CNC(C1(C)CCN(C)C1)=O)=O C12(CCOCC1)NC(=O)c1occc1CN2.c1(C(CC)COC)ccncc1 C1(NC(C(C)OCOC)=O)CCCN(C(=O)CCN2CCC2)C1 C1(C(=O)NC(C)C(N)=O)CN(C(c2cn(C3CC3)nn2)=O)CC12CC2 c1(CC(=O)NC(=O)CC2CC3CC3C2)cccnc1F.C1CCC12CC2 c1(OC)cc(C(=O)NCC(O)CCNC(=O)CSC(C)(C)C)c2ncccc2c1 CCCCCC(O)CNC(C1CCC2(CC2)N1C(=O)C(C)(C)COCC)=O O=C(N=c1cc(C2CC2)[nH][nH]1)Nc1cccc(C2(F)COC2)c1 N1(C(C(CC)CCOC)=O)CC(C)(C)OCC1CNC(=O)CC(C)(C)C1CC1 C=CC(CC)CC(=O)NCC1(CO)CCN(C(=O)CCCCC2CC2)C1 c1(N(CC(=O)OC)CC)ccc2cccnc2c1.c12ccc(cc1)oc2=O Cc1nnc2n1CC(NC(N1CC3CC4CC3C1C4)=O)CC2 C1(CNC(=O)COCCC2CCCC2)CC2CCCC2C1.C12CC(C1)C(=O)NC2 C1(NC(c2cc(C)on2)=O)CC2(C1)CC(C(N1C(C)CCCC1C)=O)C2 C(=O)(CC(C)(C(F)F)N(C)C)NC1CC(NC(c2c(C)scn2)=O)C1 Cc1nc(CC(=O)NCCCC2(NC(c3ccn(CCO)c3C)=O)CC2)c(C)s1 N1(C(C(C(=O)OCC)(C)C)=O)CC(NC(=O)C=CC2CC2)C2(CCOCC2)C1 c1(N2CCC(C)(C)C(CNC(=O)C=C3CCCC3)C2)nc2cccc(Br)c2o1 Cn1nc(C2CCC2)cc1C(=O)NCCCCNC(=O)CC1(O)CCC1 C(=O)(CCS(=O)(=O)N(C)C)NCC(CNC(C(C)Oc1ccc(C)cc1)=O)F C1(OC)CCN(C(=NCCF)NCCOc2ccc(Cl)c(Cl)c2)CC1C C(CN=c1[nH]c(Cl)c(C#N)s1)(c1ccc(C(F)F)cc1)NCC1C2(CC(C)(C)C2)C1 CCC(CC(=O)NCCCN1CCCC1)NC(C1COCC(C)O1)=O N1(C(C2(F)CCN(C(Cc3c(C)cccc3)=O)CC2)=O)CC2CCC(C1)N2C C(c1ccccc1OC(F)(F)F)=CC(=O)NCC(COC(C)(C)C)O c1(NCC2(NC(C(CC)OC)=O)CCC2)ncnc2c1ncn2C1CC1 CC(C)CCCOC(=O)NC1CN(C(c2cnc(N3CCOCC3)s2)=O)C1.C1CC1 c1(C(CC)NC(c2ccccc2)C(=O)Nc2ccccn2)ccc(OC)cc1 C(=O)(N=c1ccn(C)[nH]1)C12CC(C1)C(=O)N2.Cc1cncc(-c2cn[nH]c2)c1 c1(C(=O)NCCCCCCNC(C2C(C)(C)C2(F)F)=O)ccc(Cl)cc1N c1(C(N2CC(O)(C(C)NC(CCSc3nc(C)[nH]n3)=O)C2)=O)cn(C)[nH]c1=N c1(C(=O)NCC2(C(=O)NC(c3cncn3C)C)CC=CC2)cc2cnccc2[nH]1 C1(C)(NC(C=C2CCN(C)CC2)=O)CCCN(C(C2CCN(C)C2=O)=O)C1 CC1CN(C(=O)C(C)NC(N)=O)CCN1C(c1ccc(CN2CCC2)o1)=O C1(C(=O)NCC2(NC(C34CCC3CC4)=O)CC2)CCS(=O)(=O)C1 N1(C(C(C)NC(C2CCCC2)=O)=O)CCC(NC(c2ccc(Cl)[nH]2)=O)C12CC2 N1(C(C(c2c(C)noc2C)C)=O)CCC12CN(C(C1(C#N)CCCC1)=O)C2 Cc1ccc(F)c(C(c2nnnn2CC(F)F)Nc2cc(CO)nc(Cl)c2)c1Br Cc1cc(=N)[nH]cc1C(N1CCCC(C(=O)NC2CCC(C)(C)CC2)C1)=O C1(C(=O)NCCc2ccoc2)CC2CCCC2N1CCn1c(O)nnc1O Cn1nccc1C1=CCCN(C(=O)Cn2cnc3ccccc23)C1 C(=O)(NNc1ncnc2sc(CC(C)(C)C)cc12)C1(CC)CCC(=O)NC1=O C(=O)(C(C)(C1CCC1)NC(c1cc(Cl)ns1)=O)NC(C)CCO C(=O)(C1CCc2cccc(Cl)c21)N(C(c1ccccc1)C(=O)O)C Cc1c(C(=O)NCC(C)CNC(=O)CCc2cn(C)nn2)nnn1C(C)C C(=O)(C(C)(C)CC(=O)N1CCC(N(C(=O)CC2CC3(CC3)CO2)C)CC1)OC CC(C(=O)N1CC(F)(F)CC1CNC(C1CC1(C)C)=O)S(C)(=O)=O c1(CNCC2C(CC)CCC2)cc(OC)cc(OC)c1 C(=O)(C(C)(C)CC(C)C)NCCCCC(C)NC(C1CC(CC)C(=O)CC1)=O C1(NC(C(C)OCCN(C)C)=O)CN(C(=O)CC2CCCC(F)(F)C2)CC12CC2 C(=O)(CC(C)C(C)(C)C)N1CCC(C)(CNC(c2cnc(C(C)O)s2)=O)CC1 C#Cc1cc(C(N2CCC2(C(=O)NCC(C)(O)C(C)CC)CC)=O)ccc1C c1(CN2CCC(C(C#N)C#N)CC2)ccc(Cl)c(I)c1 C1(C(N(CC(C)OC)C)=O)CC(F)(F)CN1C(c1cnccn1)=O c1(C(=O)N=c2ccn(CCF)[nH]2)cn2cc(Cl)cnc2n1 c1(C(N2CC(O)(C(C)NC(=O)C=CC3CC3)C2)=O)c(F)ccc(F)c1Cl c1(C(=O)NCC)c(C)nn(C)c1OC1CCN(C(CC=CCC)=O)C1 c1(C(=O)NCCCN(C(c2cc(OC)cnn2)=O)CC)cc(Cl)c(Br)cn1 c1(C(N(CC(CNC(C(C(C)C)(C)O)=O)O)C)=O)ccc2c(c1)CN(C)C(=O)N2 c1(OC)nc(C)c(Br)cc1C(=O)NC(C)CNC(C1CC1C(=O)OC)=O N1(C(C(C2CN(C(=O)Cn3cccnc3=O)C2)OC)=O)CCn2ncnc2C1 C1(CNC(COCCCOC)=O)CN(C(=O)C(N2CCOC2=O)C)CC1C(F)F C1(C(=O)NC(C2(C(=O)N(CCCC(C)(F)F)C)CC2)C)CC(O)CN1C S(=O)(=O)(CCCCS(=O)(=O)NC12CCCC1C(=O)C2)NCCOC(C)CO C1(C(=O)NCC(C)OC)CCC2(CN(C(c3ccc(C)nc3OC)=O)C2)O1 c1(OC)ccc(C(N2CCCC3(CNC(=O)C4=COCCC4)CC23)=O)cc1OC C1(F)(CNC(c2ccc(Cl)s2)=O)CN(C(=O)CCOC2CCCOC2)C1 C(=O)(C1Cc2ccccc21)N1CC(O)(CNC(c2nc(C(C)(C)C)oc2)=O)C1 c1(C(=O)NCCCCNC(CC2CC(CC)C2)=O)cc2[nH]c(C(=O)OC)cc2o1 C1(CNC(CC2(SCC)CC2)=O)COCCN1C(C1CCC(F)C1)=O c1(OC)ccc(C(=O)NCCC(C)NC(C2(F)CC=CCC2)=O)cc1OC CCCCCCC(=O)N(C)CCN(CCCCCC)C(=O)Cc1c(F)cccc1F N1(C(C(CC)C(=O)OC)=O)CCC2(CC1)C(NC(=O)C(C)CF)CS2(=O)=O C1(N(C(=O)CC2(O)CC2)C)CCN(C(C2(n3cccn3)CCC2)=O)C1 C1(NC(N2CC(C(=O)OC)(CF)C2)=O)CC=CCC1C n1(CC)cc(C(N2CCC23CN(C(C2CC2c2cnn(C)c2)=O)C3)=O)ccc1=O c1(CC)cc(C)ccc1C(N1CCC(C)(NC(=O)CCCCN(C)C(C)C)C1)=O Cc1c(C(=O)NC2(CO)CCN(C(=O)CC3C=CCC3)C2)ccn1C(C)C C1(NC(C(C)OCCCC)=O)CCCN(C(=O)Cn2nccn2)C1 N1(C(C)=O)CCCCC1CC(=O)N(CCCN(C(=O)Cn1cnccc1=O)C)C c1(C(=O)NC(CCNC(Cc2c(C)cco2)=O)C)cc(Cl)c(Cl)[nH]1 c1(CNC(c2nccs2)C)ccc2c(c1)C(C)CN2C(=O)OC(C)(C)C C=C(C)CC(C)C(=O)NC12CC(NC(=O)CCc3cccc(C(F)F)c3)(C1)C2 C#Cc1cnc(C(=O)NCCc2cc(C(=O)NCC(F)CO)no2)c(C)c1 c1(C(C)(C)C)ccccc1CN(c1cc(NC(=O)C(F)OC(F)(F)F)ncn1)CC C1(c2c(C(=O)OC)c[nH]n2)CCCN(C(=O)C(=O)NC(=O)OCC(C)(C)C)C1 c1(OC)ccc2nc(N3CCCC(C)(C)CC3)[nH]c(=NCCC(=O)NC)c2c1 c1(-c2c(C(=O)NCC(C)(C)NC(C(C)NC(C)=O)=O)cno2)cccc(Cl)c1Cl c1(CC)ccsc1C(=O)N(CC(=O)N(C1CC(CO)C1)C)C1CC1 c1(C(=O)NCC2(O)CC(NC(C(CCC#C)O)=O)C2)[nH]c2c(C)cccc2c1C c1(CC(=O)NCCN(CCC)C(c2csc(C3CCCCC3)n2)=O)cncn1C C1(C(=O)NCC(C)(C)CNC(=O)CS(C)(=O)=O)COCCN1C1CCCC1 c1(N(CC(c2cccc(C)c2)C)C)nc(=NCCC2CC2)[nH]c2cc(F)ccc12 C(=O)(CC1=CCOCC1)NC1CC(CNC(C2CCC(C)(C)O2)=O)C1 C(=O)(C(CC(C)CC)NC(c1ccc([N+](=O)[O-])[nH]1)=O)N(CCCN(C)C)CCC c1(C(N2CC(NC(c3cn(CC)nc3)=O)C(C)C2)=O)cc2nc(C)[nH]c2cc1F CC1CC(C(=O)NCC(=C2CN(C(C3COC(C)(C)C3)=O)C2)F)=NO1 c1(C(=O)NC(CNC(C2(CC)CCNC2=O)=O)(C)C)cc(OC)c(C)c(OC)c1 C(CCN=c1[nH]ncs1)NC1CCN(C(COCCN(C)C)=O)CC1 c1(OC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2csc(C)c2)nc1OC N1(C(c2c(C)onc2Br)=O)CCC(C2CCN(C(=O)C=C3CCC3)CC2)CC1 N1(C(C(C)OC)=O)CCCC2(C1)C(NC(=O)CCc1cnn(C)c1)CCN2C C123CCCC1N(CCC2)C3=O.Cc1nc(-c2ncc(-c3ccccc3)o2)cs1 CC1C(C(N2CC3CCC(C2)N3C(C2CCCCC2)=O)=O)C(O)C(=O)N1C N1(C(CN(c2ccncc2)C)=O)CC2(CC(NC(=O)CC3CC(=O)NC3=O)CO2)C1 C1(N(C(c2cnc(COC)s2)=O)C)CCCN(C(C2(CF)CC2)=O)CC1 CC1CCC(CNC(=O)Cc2cc[nH]n2)CN1C(c1cc(Cl)c(Cl)[nH]1)=O N1(C(CC=CC=C)=O)CC(C(=O)Nc2ccc(Cl)c(CO)c2)C(C2CC2)C1 Cc1cc(N2CC(CNC(=O)CC3CC3C)OC(C)(C)C2)n2ncnc2n1 CC1CC(NC(=O)C(F)n2ccnc2)CCN1C(=O)COCC1CC1 C(=O)(C1=NOC2(CCC2)C1)N(C1CN(C(C2(C)COC(=O)C2)=O)CC1(C)C)C N1(C(c2n(C)nc(Br)c2)C(=O)NCCNC(N)=O)CCOCCC1c1ccccc1 c1(SC)c(F)cccc1F.c1(CC)cc(C(=O)NCC23CC(CN2C2CC2)C3)nn1C C#CCC(C)(C(=O)N1CCSC(C)(C)C1)NC(=O)C(C)NC(N)=O C1(=CC(=O)NC2CN(C(Cc3c(SC)cccc3)=O)C2)CN2CCC1CC2 CCC(C(=O)NC1(CNC(C2(CF)CC(=O)C2)=O)CC1)N1CCCC1=O C=CCCC(O)CNC(=O)C(F)CC1CN(C(C2(CCCC)CC2)=O)C1 C=CC(CCC)CC(=O)N1C(CNC(c2ccc(CN(C)C)cc2)=O)CC2CC12 CC(O)(C(=O)N1CCCC(F)(CNC(c2cnc(C(F)F)nc2)=O)C1)C(F)(F)F c1(CC(C(=O)NCCC2CC2C)NC(c2c(CC)c[nH]n2)=O)ccc(Cl)cc1Cl C(c1cc(OC)ccc1OC)=CC(=O)NCC(CC=C)NC(c1cc(CO)on1)=O N1(C(C(CC)N(C)C)=O)CCC(O)C(NC(C2CN(S(N)(=O)=O)C2)=O)C1 c1(C(=O)NCC(CNC(CC(COC)C)=O)OC)cc2sc(Cl)cc2s1 C1(C(N2CCCCC2)=O)CC2(CC2)CN1Cc1ccc(Cl)cc1C(=O)O S(=O)(=O)(c1ccc(NC(C2CCC2)C2CCC2)nc1)NC(C)CC#N C12(NC(c3c(NC)scn3)=O)CCC(CC1)N(C(=O)C(C1CC1)OC)C2 c1(OCCNC(C2CN(CC)C(=O)C2)=O)cc(Cl)cc(Cl)c1 C1(NC(C(n2c(C)ccn2)C)=O)CC2C(NC(=O)CC3COC(=O)N3)C2C1 c1(C(N2CC3(CN(C(C(C(C(C)C)O)C)=O)C3)C2)=O)cn2cccc(Br)c2n1 Cc1nccc(C(N2CCC(C)C(CC(=O)NC3CCN(C)CC3)C2)=O)c1N N1(C(C(=O)Nc2ccc(OC)cc2OC)C2CC2)CCC2(CCCCO2)CC1 C1(C(=O)NC(CC)(C)CCNC(c2cnsc2)=O)CC2C=CCC(C1)C2 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCc1cc(F)ccc1Br C(C(CC(C)C)C(=O)N1CC(F)(CNC(C2CCCN2c2nccs2)=O)C1)OC N1(C(c2c(OC)oc(C)n2)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC(C)(F)C1 C1(COC)CN(C(=O)C#CCNC(=O)CC2CC(O)C2(C)C)C1(C)C C=CCCC(CC(C)C)C(=O)NCC1CCCN(C(=O)C2=NNC(=O)CC2)CC1 Cc1nc(N2CC3(CCCC3NC(C3CC=CCO3)=O)C2)cc(C#N)n1 Cc1cc(C)n(CCCNC(=O)NCc2ccc(CO)cn2)c1 CC1=C(C(=O)N2CCCC(N(C)C(c3cccc(F)c3)=O)C2)CC1 CCCCCCC(C)(C)C(=O)N1CCN(C(c2n[nH]cc2C)=O)C(C)C1 C(CC(C)(C)C(=O)NCC(=O)NC(C1CCCN1c1nc(C)ns1)C)OC C1(C)(C(=O)NCC2CC(CNC(C3(COC)CCCO3)=O)C2)CCC2CC2C1 C(=O)(C(F)(F)c1nccn1C)N(CCOC)CCNC(=O)C(C)C1CCOC1 C1(N(C)C(c2cc(O)nn2C)=O)CN(C(C2CCC(=O)N2C)=O)CC12CC2 c1(NC(C(CC=C)C(=C)C)=O)ncnc2c1cnn2-c1ccccc1OC N1(C(C2CCN(C)C2)=O)CC2(CCC2)CC1CNC(c1cccn2cnnc12)=O C(CN=c1[nH]nc(C(F)F)s1)(C1CC1)NC(=O)Cc1cnc(O)nc1O c1(CN(C(c2nnc(C)s2)=O)C)ccccc1CNC(C1CC(O)CN1C)=O C1(C(=O)NCCC2N(C)CCC2)CN(C(=O)C(N)=O)CC12CCC2 N1(C(C(C)SCCCC)=O)CC2CC(C1)N2C(c1ccc(C)n1C)=O CC1CN(C(=O)CC2(C)CCOCC2)CC(C)C1NC(c1cc(F)n(C)n1)=O C(CCCCC(=O)NC(C)CCCC(=O)NC1(CO)CC(C)C1)=CC N1(C(C(COCC=C)C(C)(C)C)=O)Cc2ccc(Br)cc2OC2(CCC2)C1 N1(C(CSCC(C)C)=O)CCOCC(F)(CNC(c2nnn(C)c2C(F)F)=O)C1 N1(C(c2nc(OC)oc2)=O)CC(OC)CC(NC(c2cnoc2C(C)C)=O)C1 Cc1ccnc2c(C(N3CC(CNC(c4coc(Cl)c4)=O)CC3C)=O)cnn12 C(=O)(CCC(=O)NN(C)C)N1C(C)CC(NC(CCSCCCC)=O)C1 C1(NC(C(C2CCOCC2)C)=O)C2COCC1CN(C(c1ccnnc1)=O)C2 CCC(CC)C(C(=O)NCC12CCC(CC1)N2C(=O)C(O)C(F)(F)F)OC c1(OC)ccc2cnc(N(c3ncnc4c3cnn4C)C3CC(N)C3)nc2c1 C1(C(N2CCC(NC(COC)=O)C2C(C)(C)C)=O)CC(C)(C)OC(C)(C)C1 C1(C(N2C(C3(C(=O)NCCS(CC)=O)CC3)CCC2)=O)CCCOC1C Cn1nc(C(C)(C)C)cc1NC(c1cncc(C(N2CCCCC2C(N)=O)=O)c1)=O C1(C(=O)NCC)CCCN(C(=O)C(c2ccc(Br)cc2)OC)C1C CC1CN(C(C2CCCNS2(=O)=O)=O)CC(C)N(C(=O)CCC2(O)CCC2)C1 c1(SC)nc(Cl)c(CNC2C(F)(F)CCN(C(c3ccc(O)nc3)=O)C2)c(Cl)n1 C1(CC)CCCNC1C(=O)NCCC(=O)NCC1CC1 C(=O)(C#CC1CCOC1)NC(CC#C)(C)C(=O)NCCC12CCC(CC1)C2 C(=O)(CC(CC)(C(F)F)NC(C)=O)N1CCC(c2ncc(C)cc2C)C1 N1(C(C(CC)=CC)=O)CC(C)N(C(=O)COC2CN(C(=O)CC)C2)CC1C CCC(O)CC(=O)N1CCC(C(=O)NC2CC(F)(F)C2)(CF)C1 N1(C(=O)CCSC2CC2)CCCC(Cc2ccc(O)nc2)C1 Cc1cc(=NC2CC(N3CCCC3)C2)[nH]c(=NCCCN2CCC(C)CC2)[nH]1 C(C1=CCN(C(c2csc(-c3ccccc3F)n2)=O)CC1)NC(CCOCC)=O c1(OC)ccc(CNC(=O)C(c2cn(C)nc2C)N(C)C(C)C)cc1 c1(CC)nc(C)oc1C(=O)NCCC(O)CNC(=O)CC(c1ccccc1F)C c1(-c2nc(CC)on2)cccc(C(=O)NC)c1.C1(CN2CCN2C)CCOCC1 C(C1c2ccsc2CCN1C(=O)C(C)CC(C)COC)NC(CC=CC=C)=O C1(CC)(CNC(=O)CC2SCCN2C(=O)OC(C)(C)C)CCCN(C(C)=O)C1 C1(C(=O)NCC(CC(=O)NCc2nocc2C2CC2)OC)CC(C(C)C)=NO1 Cc1nc(Cl)[nH]c(=NC2CCCC3CN(C(C4(O)CC4)=O)CC23)c1[N+](=O)[O-] c1(C(=O)NCCC(=C)CNC(c2nnc(S)n2C)=O)c(C)ccc(C)c1N C1(NC(CCC(=O)OC(C)(C)C)=O)CCCCCN(C(C2(CO)CCC2)=O)C1 C#CCCCCCC(=O)N1CCC(NC(=O)CCN2CCCCCC2)C1 C=CCC(CC=C)C(=O)N1CCCC1CCNC(C1CCCN1C1CC1)=O C1(C2CCCC2)(C(N(C(C)CNC(C2CCCN2N=O)=O)C)=O)CCC1 C12(OC)CCCC(C(=O)Nc3ccc(-c4nc(CN)no4)cc3)(CC1)C2 c1(C(N2CC(CCNC(c3conc3C3CCCC3)=O)C2)=O)nsnc1O CCCCCC(C)(C)C(=O)NC(C1CN(C(=O)C(CC)c2ccccc2)C1)C C(CC(C)C)(C(=O)NCC(C1CC1)N(C)C(C1(c2ccccc2Cl)CC1)=O)OC CC1=C(C(=O)NCCC(O)CNC(=O)CC2CN(C)C2)SCCO1 CC1(C)CCN(C(c2cccc3c2COC3)=O)CC1NC(=O)CC1=CCCCC1 C1(OC)CC(F)CN(C(=O)CC2CCC(NC(=O)CCCN=[N+]=[N-])CC2)C1 C1(NC(C(CN(CC)CC)F)=O)CCN(C(=O)CC2CC(C)=NO2)C1(C)C c1(C(N(CCCCNC(C=CC(CC)C)=O)C)=O)cc2cccc(N)c2cn1 c1(CNC(c2cccc(-c3ncco3)c2)C)ccc(N)cc1[N+](=O)[O-] N1(C(c2c(C)n[nH]c2C)=O)CC2(CCCCN(C(C3(C)COCCO3)=O)C2)C1 CCCCCCC(C)(CC)C(=O)N1CCCC(CN(C(=O)C(C)SC)C)C1 N1(C(C2C(=C)CC2)=O)CCCC(N(C)C(c2cccc(CNC(C)=O)c2)=O)CC1 C=CC(C)(CCOC)C(=O)N1CCCC(NC(=O)C(C)C(=O)OC)C1 N1(C(C2CCC(CC)CC2)=O)CCCC(CNC(=O)COC2CC=CC2)(OC)C1 C1(C#N)(CCC(N2CC(CNC(=O)OC(C)(C)C)C2)=O)CCC1 CCCCCC(=O)N1CC(CC)CC1CNC(C1CC1CCOC)=O C1(C(=O)NCC2(NC(c3nnc(C(C)C)s3)=O)CCC2)Cc2ccccc2CO1 CC1CN(C(C2CCSCC2)=O)CC(C(=O)NCC2(C)COCCO2)O1 C1(C(=O)NCC(C)CN(C)C(c2ccncc2F)=O)CC12CCCCCC2 C(C)(CCC(=O)NCC1(CNC(c2ccc(N)cn2)=O)CC1)OC C1(c2nnnn2C2CC2)CCC(F)(F)CC1.O=C(O)C(C(=O)NCCCl)C1CC1 C=CCCCCCC(=O)NCC(c1ccccc1)NC(=O)C=CC1CC1 c1(C(N2C(CNC(C(C=C)O)=O)CC(OC)C2)=O)cccc(F)c1Cl CC1C2CCCCC2CN1C(=O)CN(C1CCC1)C(C1CCC(O)CN1C)=O C(=O)(C(N)CC(C)(F)F)N(C)CC(C)NC N1(C(C2C(C)(C)C2)=O)CC(NC(c2cccc(P(C)(C)=O)n2)=O)CC12CCOC2 Nc1c(O)ccc(Cl)c1C(N1CC2C(CNC(C3CCCN3C=O)=O)C2C1)=O Cc1cc(C(N2CCC2CNC(c2ccn(C3CCOCC3)n2)=O)=O)n(C)n1 C1(C(N(CCCCNC(=O)CC2CCS(=O)(=O)C2)C)=O)C(F)(F)C12CCC2 n1(CC)cc(C(=O)N(C)CC2CCCN2C(C2CC2CF)=O)cn1 CN=c1ccc(C(N2CCCC(CNC(=O)C=C3CCC(C)C3)CC2)=O)c[nH]1 CC1CN(C(=O)C(n2cc(Cl)cn2)C)CCC1NC(=O)C=CC1CCOCC1 N1(C(c2cc(CC)no2)=O)CC(NC(C2Cc3nccn3C2)=O)CC(C)(C)C1 C1(NC(C2(CC)CCOC2)=O)CC2CC(C1)N(C(=O)Cc1cccc(Cl)c1F)C2 CC1CN(C(C2CC(C)C2)=O)CCC1CNC(c1ccc(C(C)(F)F)cc1)=O N1(C(CCCOC(C)C)=O)CC=C(C(=O)N2CC(CO)C(C)(C)C2)C1 n1(COC)nccc1C(N1CCC(CCC(=O)NCC(=O)OC)C1)=O c1(C(N2C(C(=O)NC3CCN(C(C)=O)CC3)CC(=C)C2)=O)c(Cl)ccc(Br)c1Cl Cc1nc(C(C)C)nc(O)c1C(=O)NC1CCN(CCCCCF)C1 CCC(C)(CNC(c1cn(CCO)nn1)=O)C(=O)NCCC1(C)CC1 C(C1CCOC1)=CC(=O)NCC(C)CN(C(=O)C=CSc1ccccc1)C c1(C(N(CCNC(CN2C(C)CC2)=O)C2CC2)=O)cccnc1S c1(C(=O)NCC23C(CN(C(c4c(Br)c(C)n(C)n4)=O)C2)C3)ccc2ncnn2c1 N1(C(CN(C2CC2)CC)=O)CCC2CC1CN2C(C1OCCC1C(F)(F)F)=O c1(CN(C(C(N2CCC(CC)C2)=O)=O)C)ccc2[nH]c(C(=O)O)c(C)c2c1 C1(C(N(C2CC(NC(C3(C)CCC3)=O)C2)C)=O)CCC(=O)N(c2cnn(C)c2)C1 c1(OC)cc(NC(c2csc(-c3cnn(C(C)C)c3)n2)=O)ccc1CN(C)C C(=O)(C#CC1CCCCO1)NC1(CCCNC(CN2CCN(C)C(=O)C2)=O)CC1 c1(-c2cn(CC(=O)NC3CCC(C)C3C)nn2)ccc2cc[nH]c2c1 N1(C(c2cccc(C)n2)=O)CCCC2(CCC(NC(c3ncn(C)c3C)=O)C2)C1 C1(C)(NC(CC(CC)OC)=O)CCCCC1C(=O)NC1CCCC1C#N C1(C2CN(C(=O)C(F)CC(C)C)C2)(NC(c2c(C)nsc2)=O)CC1 C(=O)(C1=CCOC1)NC(CC=C)CNC(=O)CC1CCC(=O)N1 C1(CNC(Cc2cc(C)ns2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C CC(CCc1cn[nH]c1)N=c1nc(N(C)CCC2CC2)c2ccccc2[nH]1 C1(NC(CN(C(C(C)C)=O)C)=O)COC2(CCCN(C(C3(C)CSC3)=O)C2)C1 CC1CCN(C(c2cc(O)ncn2)=O)C1C(=O)NCCN1CC2CC2C1 c1(C(N2CC(NC(CCC#CC)=O)C(CO)CC2)=O)cc2ccccn2c1 O(NC(=O)C1CC(SC)C1)CCCOC.C1C(CO)NC(=O)N1 C1(C(N2CCN(C(=O)C(O)C(F)F)CC(O)C2)=O)Cc2cccnc2C1 C=C(C)CCC(C)NC(=O)CCC1CCC(NC(=O)C(C)N(CC)CC)C1 C=Cn1nccc1C(=O)N(C)CC1CCCN1C(C1(OC)CCCOC1)=O CC1(C(=O)NCC2CN(C(=O)CCNC(N)=O)CC2C(F)(F)F)CC(C#N)C1 C1(C(=O)NCC2(O)CCN(C(=O)CSCc3ccncc3)C2)CC2CC1C1CC21 N1(C(C2C(OCC)C2)=O)CCC(C2CC2)C1CNC(=O)C(F)C(C)C c1(N2C(=O)CC(C(=O)N(CC(F)F)Cc3ccccc3)C2)cc(F)cc(F)c1 n1(CC)nc(C(=O)NCc2cccc(NC(c3ccncc3Cl)=O)c2)ccc1=O CC(Cc1cnc[nH]1)C(=O)N(CCCCNC(=O)C(C)(C)c1ccc(Cl)s1)C N1(C(=O)Cc2ccon2)CCC(N(C(c2cncnc2)=O)CC2CC2)C12CCC2 c1(C(=O)NCC2CC(CNC(CCC(=O)NCCC)=O)C2)cc(C)nc(C)c1 Cc1c[nH]c(C(=O)NC2COCC2NC(=O)CCC2CCN(C)C2)c1 CCC(CCC(=O)NC(c1nccs1)C)NC(c1ncncc1Cl)=O c1(C(=O)NC2C(NC(C(CN(C)C)O)=O)COC2)cc(NC2CC2)ncc1Cl c1(C(C(=O)NC2CC(NC(c3cn(CC)nn3)=O)C2)(C)F)ccccc1F CC1(CNC(=O)Cn2nnc(C3CC3)n2)COCCN(C(C23CCC(C2)C3)=O)C1 CCCCC(F)(F)C(=O)N1CC=C(C(=O)NCC(O)CCC)C1 OC1CCCC2CN(Cc3cccc4ccoc34)CCC12 C12(NC(C(C)n3cccn3)=O)COC(CNC(C3(C#N)CC3)=O)(C1)C2 c1(NCC(C)NC(C(=O)NCC)=O)ccc2c(c1)CCC(=O)N2CC CN1CCC(CN(C(c2csc([N+](=O)[O-])c2)C(=O)NCC(F)F)C)CC1=O c1(C(N2CCC(n3cc(CNC(CSC)=O)nn3)C2)=O)cc(C)ncc1Cl C1(C(C)CNC(=O)CSC2CC2)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1 C1(NC(CC(C)C)=O)C(CNC(=O)CC2CC2C)CCC12CCC2 C1(C)(C(=O)NC(C(=O)NCCCCC)COC)CC2CC2C1 CC1CN(C(=O)CCC2CCC2)CC1CCNC(c1ccsc1)=O C1(C2CN(C(=O)C(=Cc3c[nH]cn3)F)C2)(NC(=O)C=CCOC(F)(F)F)CC1 c1(CC)nc(C)c(C(=O)NCC(F)CNC(C2CC(O)(c3ccccc3)C2)=O)s1 N1(C(C2(CCOCC)CCC2)=O)CCCC2(C1)CN(C(=O)C1=NNC(=O)C1)C2 c1(-n2c(Cc3nc(C)ccc3F)nc(CC(C)OC)n2)ccc2nn[nH]c2c1 O=S(=O)(c1cccnc1NCC1CCCOC1c1cn[nH]c1)NCC1CCOCC1 c1(C(N2CCC(c3ccc(C#N)s3)C2)C(=O)NC(C)C)cnn(C)c1F C#CCC(C(=O)N1CCCC(NC(=O)C(C#N)C#N)C1)C1CC1 N1(C(c2c(C)nc(O)cc2)=O)CC2(CCN(C(C3CC3CC(C)C)=O)C2)C1 CC(C)C(CC1CCCC1)C(=O)Nc1ccc(C(O)Cn2ccnc2)cc1 n1(CCC(=O)NCC(C)NC(=O)C=CC(=O)OC)c(C)csc1=O.C(COCCO)OC C(=O)(CCC(C)CCCC)NCc1c(C(=O)NC(CC#C)CC(=O)OC)con1 C1(C)(CC)CCC(C(=O)NC(C)(C)CNC(c2cc(C3CC3)nn2C)=O)O1 O=C(O)C1c2ccccc2CCN1Cc1cnn2c1OCCC2 CC1CN(C(c2c[nH]nc2C(F)F)=O)CCC1NC(C1(F)CCOC1C)=O Cc1coc(C)c1NC(N1CCC1c1cn(C2(OC)CCOC2)nn1)=O C1(C(=O)NC(CCCNC(c2c(C)nco2)=O)(C)C)OCC2COCCC12 C1(CNC(c2cnc(CC)[nH]2)=O)CCC(NC(=O)Cc2cnc(C3CC3)[nH]2)CC1 C1(C(N(CCCNC(=O)C(F)(F)C2CCCC2)CC)=O)CC1C1CCCC1 CC(CC1CCCCC1)N(C)N1CCCC(C)C(F)(F)C1 C1(NC(c2c(OCCC)cccc2)=O)CCN(C(c2ncc[nH]c2=O)=O)CC1C C1(C(=O)NC(CC)CN(C(=O)C=CC(C)(C)C)C)CCC(=O)N1C C1(CN(C(CSCC=C)=O)C)CCCCN1C(=O)Cc1sccc1C N(C1CCc2cc(CNC(C3(C)CCC(C)(C)CC3)=O)ccc21)C(C=CSC)=O c1(C(N(CCCNC(C2ON=C(C)C2)=O)C(C)C)=O)ccc2nn[nH]c2c1 c1(NC(C23CC(=O)C2CCC3)=O)ccc(Br)c2c1CCC2 Cc1ccc(N(C)C2CC2)c(C(=O)Oc2ccc(C)cc2C)c1.C1C=CC1 C(=O)(C(C)(O)C(C)C)NCC(C(=O)NCC(C)(C)N(C)C)OC c1(C(=O)NCC2(C(=O)NCC(N(OCC)C)=O)CC2)n[nH]c2ccccc12 O=C(NN1CCCC1C(=O)NCC1CCCCC1(F)F)c1cnns1 n1(CC)cnc2c(N3CC4C(C3)C4(C)C)nc(=NCCCC#N)[nH]c12 N1(C(c2coc3c2CCCC3)=O)CCCC1C1CCCN1C(c1cc[nH]c1)=O C(CC1CC1)(C(=O)NCC1CCCS1)NC(C1(CC=C)CC1)=O CCC(CN(C)C)CC(=O)N(C)CCN1CCN(C(=O)C(C)N2CCCC2)CC1 CCC(C)C(CC(=O)NCC1CC12CCCCC2)NC(c1cc(C)oc1CC)=O c1(C(=O)NC2CN(C(C3(F)C(C)C3)=O)C2)ccnc(N2CCOC(C)C2)c1 c1(C(N2CC(NC(c3c(C)cc(F)s3)=O)C(C)C2)=O)ccc(Br)cc1F c1(C(=O)NC2C(C)N(C(c3ccsn3)=O)CCC2)cc2c(=O)[nH]ccn2n1 C(=O)(C(C)CCC(C)(C)C)NC1(CNC(C=CCCC)=O)CCOCC1 C1(NC(Cc2c(C)cco2)=O)CN(C(=O)CN2CCC(N(C)C)CC2)CCC1C N1(C(C(C2CCC2)OC)=O)CC(F)CC1CN(C)C(c1cc(C)ns1)=O C1(OC)CN(C(c2cc(Cl)cn2C)=O)CCC1NC(=O)CC1CCCC1(F)F c1(C(=O)NC(C(C)NC(c2c(C#C)cnn2C)=O)C)cc(Cl)c([N+](=O)[O-])[nH]1 C(CN=c1[nH]c2cc(Cl)ccc2s1)OCCNC(c1cc(O)nc(Cl)c1)=O N1(C(C)=O)CCC(Cn2cc(-c3cccc(CO)c3)nn2)C(CO)C1 c1(NC2C(C)CN(C(C(C)(C)OC)=O)CC2C)ncnc2[nH]c3ccccc3c12 N1(C(Cc2nc(C)sc2)=O)CCCC2CN(C(C3(CO)CCCC3)=O)CCC12 c1(C(N2C(C(C)NC(=O)CC3CC3(C)C)CCC2)=O)nnn(C)c1C(F)(F)F c1(C(N(C2CN(C(=O)CC(OCC)OCC)C2)CC#C)=O)cc2cccnc2cn1 c1(C(=O)NCC(CCNC(C(C)c2ccsc2)=O)O)cn2ccc(F)cc2n1 c1(C(=O)NCC2CC(NC(C(C)CC3CC3)=O)C2)ccc(-c2ncc[nH]2)nc1 CC(C)C(CN(C)C)C(=O)NCCCCNC(C1(O)CCOC1)=O C1(C(=O)NC2CC(NC(C(C)CC3CC3)=O)C(O)C2)CC2(CCCC2)C1 n1(CC)nc(C)c(C(=O)NC2CCCC2CNC(=O)CN2CCCC2=O)c1Cl CCC(CN(C)C)C(=O)N1CCCC1CCNC(c1c(C)ncn1O)=O c1(C(=O)NCC2(O)CN(C(=O)CC3CCCCC3)C2)cccn(C2CC2)c1=O C1(NC(=NCCOCC)NCCOCC(C)C)CC2(CO1)CC(F)(F)C2 N1(C(Cc2c(C)scc2)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC2(CC2)C1 C1(c2nnnn2C)(NC(CC)C)CCCC(CN(C)C)C1.SC C1(CC)CN(C(C23CC(C)(C2)OC3C)=O)CCC1NC(=O)CC1C(=O)ON=C1C N1(C(C2CC3C(C)(C)C3C2)=O)CC2CCC(C1)C2NC(=O)CN1CCC(F)CC1 C1(CC(=O)N(CC)Cc2cccc(F)c2)CN(C(C)(C)C2(SC)CC2)CC12CC2 c1(CCC)cc(=NC(=O)N2CC3CCC3C2CO)[nH]n1C c1(C(=O)NCc2ccc(CNC(C(CO)OC)=O)cc2)ccn2ncc(C)c2n1 CCCC(CNC(C1CCCN1C(=O)Cc1cscn1)=O)CCC C12(CNC(c3ccc(CO)cc3)=O)CCC1CCN2C(=O)Cn1cccn1 c1(CC)occc1C(=O)NCC(CCOC)NC(c1cnn(CC(C)C)c1)=O Cc1cc(C(=O)NCC2CCN2c2ncns2)ncc1C(F)F N1(C(C(C(C)C)CN(C)C)=O)CCOC2(C1)CN(C(C1CN3CCC1CC3)=O)C2 c1(SC)ccc(O)c(C(=O)NC2CC3CN(C(=O)CCc4cn(C)nn4)CC23)c1 Cc1cc(S(=O)(=O)N2CCCC(CC(=O)Nc3ccc(O)nn3)C2)c(F)cc1Cl c1(-c2cccc(CC(=O)NCC3CCS(=O)(=O)C3)n2)c[nH]c2ncccc12 N1(C(CC)=O)CCC(NC(c2cc(C)n(C)n2)=O)C(O)C1 c1(NC(C23C(CN(C(=O)CNc4ccccc4)C2)C3)=O)ncc(Cl)cc1F c1(C(=O)NC2(CF)CCN(C(=O)C=CC=C(Cl)Cl)C2)cnc2ccnn2c1 c1(CN(C2CC3(CNC3)C2)C(c2ccccn2)=O)c(Cl)cccc1Cl N1(C(C2N(C(C)=O)CCC2)=O)C2CCC1CC(N(C)C(C1CCS1(=O)=O)=O)C2 c1(CC2(NC(=O)CC3CC3(Cl)Cl)CCCC2)ccccn1 CC1C2CCC(C2)C1C(=O)NCCC1(C(=O)N(C)CC2CC(O)C2)CCCC1 CC(C)(CCC#N)C(=O)N1C2CCC1CN(C(=O)CC1CNC(=O)C1)C2 n1(CC=C)c(N(CCF)CC2CCC2)nnc1CC(C)(C)C C1(NC(=O)NC2CC(OC)C2)CCC(n2cc(C3SCCS3)nn2)CC1 CS(=O)(=NC(=O)C1(CO)CC1)c1cnn2c1CN(C(c1ccc(CO)o1)=O)CC2 Cc1nn[nH]c1C(c1ccccc1)NC(C1COCC1NC(=O)Cn1cccn1)=O C#CCC(C)(C(=O)N1CC(c2nncs2)C1)NC(=O)CCc1ccccn1 CCC(C)(C)C(O)C(=O)NCCC1(OC)CN(C(=O)C(c2cccc(C)c2)C)C1 C1(C(=O)OCC)CCCCC1.C(C)(CNC(=O)COCCOCCO)(C1CC1)OC S(=O)(=O)(C1CC1C)NCCC(=O)N(c1ccccc1)C(C)C N1(C(C2CC3CCC2O3)C(=O)NCc2c(OC)cccc2)CCC2(CC1)CC2 C1(CNC(c2n[nH]cc2C(=O)O)=O)CCCN(C(=O)C=CCOc2ccccc2)C1 c1(C(=O)NCC2(F)CN(C(c3cnc(C4CC4)nc3)=O)C2)c[nH]nc1[N+](=O)[O-] CC(C)C(C)(C)C(=O)N1CCCC(N(C(=O)C(N2CCC(C)CC2)=O)C)C1 C1(C(=O)NCCCCNC(Cc2n(C)ccn2)=O)CCN2CCC1C2 C1(C2CN(C(c3ncsc3C(C)C)=O)C2)(NC(c2n(CCC)ccc2)=O)CC1 C1(NC(C(CCOC)C)=O)CCCC2CN(C(=O)C=Cc3cn(C)cn3)CC12 C1(CNC(Cc2c(C)scc2)=O)CCCN(Cc2cnccn2)C1 C1(C(=O)NCC(CC(C)C)NC(C2(n3cnnn3)CC2)=O)CCCC2(C1)CC2(F)F N1(C(c2n(C)ccn2)=O)CCCC(NC(=O)C(O)CCCc2ccccc2)CC1 c1(C(N(CC(=O)NCC(O)C(C)O)CCC)=O)cc([N+](=O)[O-])c[nH]1 c1(CC)cc(O)ccc1NC(C12CCC(CC1NC(=O)CCCCCF)C2)=O CC1SCCCC1C(=O)NC(c1ccccc1)C(N1CCC2CC12)=O CCCCC(O)CC(=O)N1CCN(C(c2ccnc3[nH]cnc23)=O)C(CF)C1 c1(COC)nc(C(=O)NC(CO)C(C)NC(=O)C(F)OC)cs1 C1(C)(CN(c2ccc(C)cc2)C(=O)NCCCN2CCCC2=O)CCC(O)CC1 C1(O)(CCNC(CSC)=O)CCCN(C(=O)CC2(OC)CCCC2)C1 c1(C(=O)NC2CC(C(C)NC(C3CC(O)C3)=O)C2)csc(C(C)(C)C)n1 C1(C(N(C2CN(C)C2)C)=O)(CF)CCN(C(=O)C=Cc2cnn(C)c2)C1 c1(CCC)ccc(C(C)(C)OC)cc1.C12(CCC1)C(=O)NCC1CC1NC2=O c1(C2N(C(C3CCN(CC(F)(F)F)C3)C)CCC2)ccc(Br)s1 C(=O)(CCCC(=O)N1CCCC1)N1CC(CNC(C2CC=C(C)CC2)=O)OCC1 c1(C(=O)NCCCN(C(C2(C(=O)OCC)CCC2)=O)C2CC2)cc[n+]([O-])cc1 C1(C(=O)NC(CCC)CO)CCCN(C(=O)C(C)CC#N)C1 C1(C(=O)NCCCCC=C)CCC2(CC2)N1C(C1CCCC1OC)=O N1(C(c2cn(CCC)nn2)=O)CC(CNC(=O)CN2CCCC2C)OC(C)(C)C1 n1(CC)cc(Cl)c(C(=O)NC2CC(O)(CNC(=O)CC3CCCN3C(C)C)C2)n1 CC1(C)Cc2cccc(C(N3CC4CCCC(NC(C5(F)CC5)=O)(C4)C3)=O)c2O1 N1(C(CC=CC)=O)CCC(c2cccc(F)c2)C(NC(=O)C(F)(F)CC)C1 Cc1nc(C(C)C)ccc1C(=O)NCC1(C)CCCN1C(C1CCOCC1)=O C=CCCCCCCC(=O)N(CC(=O)N(C)Cc1ncco1)C CCCCC(O)CC(=O)NC(C1(O)CN(C(=O)CSc2ccc(C)cc2C)C1)C Cc1cc(C)c(C(N2CCC(N(C(=O)C=CC(=O)N(C)C)CCO)C2)=O)s1 C1(C(NOCCOC(C)C)=O)C2CN(C(=O)CC3CC=CCN3C)CC12 N1(C(C(CCC)O)=O)CCC(C2(CNC(C3(O)COC3)=O)CCOCC2)CC1 CCCCC(C)(F)C(=O)NCC#CCNC(=O)CC1CC(CC)=NO1 CC1CCCN(C(=O)C(=O)NC2CC(N3C(=O)CNC3=O)C2)C1CO C=C(Cl)CCC(=O)N1CCCC1CN(C1(COC)COC1)C(=O)OC(C)(C)C N1(C(c2c(CCC)nns2)=O)CCC(C2CCN(C(c3ocnc3C)=O)C2)C1 C1(NC(C(COC)(C)C)=O)CN(C(c2ccnc(C(F)F)c2)=O)CCC1C c1(-c2cn(CCCNC(=O)NCCC3CC4CCC3C4)nn2)ccc2c(c1)CC2 C1(CC(=O)NC(c2nc(=O)o[nH]2)C)CN(C(=O)C(c2ccc(C)o2)C)CC(C)O1 C1(N(C(c2c(CC)nccn2)=O)C)CCCN(C(=O)COC2CCOCC2)CC1 N1(C(c2ccc(NC(C)=O)cc2)=O)CCC(NC(c2nnccc2C)=O)C(C)C1 O=C1CC(C(=O)NCC2CC(NCc3ccccc3)C2)c2cccnc2N1 C(C)(C)(CC(=O)N1CC(NC(C2CC(=O)N(c3cn[nH]c3)C2)=O)C1)OC C1(C(N2CCCC(C(=O)NCc3nnc(CC)o3)C2)=O)Cc2ccccc2C1 c1(CCN2CCC(C)(CC)C2)cccc(C)c1C n1(CC(=O)NC(CC=C)CNC(C2(CF)CCOCC2)=O)ccc(C)cc1=O C1(C(=O)NCC2(C)CC(NC(=O)C3=CCSC3)C2)CCCNS1(=O)=O c1(C(=O)NCC(N(C(=O)CC2C=CCC2)C)C2CC2)cn(C2CCCC2)nn1 c1(CC(=O)NC2CCC(C(N3CCC(O)CC3)=O)CC2)cc(Br)cc(Br)c1 C1(CC(=O)N(C)CC2CCCCN2C(c2cnnn2C)=O)CC2(CCC2)CO1 C12(NC(C(c3ccnn3C)NC(C(CCCC)F)=O)=O)CC3CC(CC1C3)C2 C1(C(N2CCCC(CCO)C2)=O)C(C2CC2)CCN1C(c1ccccn1)=O C(=O)(C(S(C)(=O)=O)C1CC1)NCCCN(C(=O)Cc1coc(C(F)F)n1)C(C)C Cc1c(Cl)ccnc1C(=O)NCC(O)CCNC(C1(C(C)C)CNC(=O)C1)=O CCC(CC(=O)NC1CN(C(=O)C(O)c2cnc[nH]2)CC1(C)C)C(F)F C(C(C(=O)NCCCc1nccs1)C(C)(C)C)NC(c1scc(C)c1)=O c1(C(=O)NC2C(CNC(c3c[nH]c(=N)o3)=O)CCC2)cc(Cl)ncc1F c1(CCC)noc(CCC(=O)NCC2CCN(C(=O)Cn3ccnn3)C2)n1 Cc1cc(C(=O)N(CC(C)O)CCn2cc(-c3csnc3C)nn2)on1 Cc1nc2cncc(C(N3CCCN(C(c4nc(O)sc4C)=O)C(C)C3)=O)c2[nH]1 N1(CC(=O)NC(c2ccccc2)C(=O)NCC2(C(=O)OC)CC2)CCOC1=O C1(NC(c2c(CC)c[nH]n2)=O)CC2CC1CN(C(=O)C(O)C(C(C)C)OC)C2 c1(C(N2C(CNC(C3CCCS3(=O)=O)=O)CC2)=O)ccc(CO)c(F)c1 CC1CCN(C(C2CC(F)(F)CCC2(C)C)=O)CCN1C(=O)CCCS(N)(=O)=O N1(C2C(OC)COCC2)C(=O)NC(C2CCN(c3cccc(C)c3C)CC2)C1=O CC1CCCC=C1C(=O)NC1(C(=O)NC2CC(C(F)(F)F)C2)CCSC1 c1(C(N(CC(C)NC(c2nccnc2C)=O)CC)=O)ccc2nsnc2c1 C1(O)(CCNC(C(C#C)(C)C)=O)CCCN(C(=O)C(CCSC)NC(N)=O)C1 C1(C(=O)NC(C2CCN(C(=O)CCn3cc(Cl)cn3)CC2)C)CCC2(CC1)CC2 c1(C(=O)NCC2CCCC(NC(c3ccncc3)=O)C2)cc2n(c1)CCC2 Cc1nn(C)c(C)c1C(C)C(=O)NC1CCCC1NC(c1cnsn1)=O c1(C(N2CCN(CCNC(c3c(COC)cc[nH]3)=O)CC2)=O)ncc(Cl)cc1Cl C1(NC(CN(C)C(c2ccsc2)=O)=O)CN(C(=O)C=C2CCSCC2)CC1(C)C c1(C(N(CCCNS(C)(=O)=O)C2CC2)=O)cn(C2CCCCC2)nn1 n1(CC)cnc2c(NCSC)nc(N3CCOC(C(C)(C)C)C3)nc12 c1(OC)ccc(C(CNC(C2(C)COC2)=O)NC(=O)Cc2ncoc2C)cc1 Cc1cnc2ccc(C(=O)NC3CN(C(=O)C4=CCCC4)C4CC34)cn12 CN1CC(NC(C2(CCNC(=O)CC3CCC(O)C3)CC2)=O)CC(C)(C)C1 N1(C(c2nn(CC)c(O)c2)=O)CCCN(C(c2sccc2SC)=O)CC1C C(=O)(C1=CNC2=NCCCN12)NC1(CC=C)CN(C(=O)CN2CCS(=O)CC2)C1 N1(C(CNC(c2ccc(C)cc2)=O)=O)CCN(C(=O)CCCCN(C)C)C(C)C1 c1(NC(C(N2CC(CCC)OCC2)=O)=O)ccc(Br)cc1OC(F)F CCC(CC(=O)N1CCOC(CNC(C2CN(c3nnnn3C)C2)=O)C1)C(C)C C1CCC2(CC1)CC2.C1(C(=O)NC2CC(CC(=O)NCC)C2)CCOC1C1CC1 c1(CN2C(C(=O)N=c3[nH]ncs3)CC(O)C2)csc2ccccc12 C#CC(C)(C)C(=O)N1CC(CCNC(c2c(C)coc2C2CC2)=O)C(C)C1 C(=O)(CC(C)(C)C(F)(F)F)N1CCC(Nc2c3cnn(CC(=O)OC)c3ncn2)C1 c1(C(=O)NCC2CN(C(c3c(OC)c[nH]n3)=O)CC2C)cc2ccncc2s1 N1(CC(N2CC(CCN(C)C)(NC(C(c3ccccc3)C)=O)C2)=O)CCCCC1C N1(C(C(CC(C)C)OC)=O)C2CCC1CN(C(=O)Cc1cscn1)C2 c1(OCCNC(C(C2CCN(C(=O)OC(C)(C)C)CC2)F)=O)ccc2scnc2c1 Cc1ccc(C(=O)NC2(C)CC(NC(c3csc(S(C)(=O)=O)c3)=O)C2)cc1C#N C(CC)(CC(=O)N1CC(CC)(CC)C1)N(C(C(CC)=CC)=O)C C#Cc1ccc(CC(=O)NCCC2CSCCN2C(=O)C(O)C=C)cc1 N1(C(C(C)c2cccs2)=O)CCOC2CCN(C(c3cnc(O)c(F)c3)=O)CC12 N1(C(c2cc(OCC)ns2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC(F)C1 C(CC(C)C)(C(=O)NCCC1(OC)CN(C(=O)Cc2cc(F)cc(F)c2)C1)OC c1(C(C(=O)C(C2CCC2)C2CCC2)C)noc(C(F)(F)F)n1.NC C1(NC(CCc2c(C)noc2)=O)CCCC(=O)C1.C12(C(C)(C)O)CN(C1)C2=O C(C(F)(F)C(F)(F)F)OCCC(=O)NC1C(NC(Cn2c(C(C)C)ncc2)=O)C1 c1(CNC(CCN(CC=C)C(c2cn(C)nn2)=O)=O)cccc(C)c1C c1(C(c2n(CCCSC)nnn2)NCC(C)OCCO)ccc(S(N)(=O)=O)cc1Cl C(=O)(CC(CC(=O)O)C1CCC1)NC(C1C(c2cn(C(C)C)nc2)C1)=O Cc1ncsc1C(=O)N(C1CC1)CC1CCCN1C(=O)C=CCF O=C(C1=C2CCN=C2NC=C1)NC1CS(=O)(=O)CC1NC(c1ccncn1)=O c1(C(=O)NCC(C)N(C)C(c2cccc(N3CC=CC3)c2)=O)cn(C)[nH]c1=N c1(C(CNC(C(CC)O)=O)NC(C2(c3ccn(C)n3)CC2)=O)ccccc1F C(=O)(C(CC(C)C)Oc1ccc(O)c(F)c1)N(CC#C)CCC N(C1CCOc2ccccc21)C(=O)CNC1CC2CC1C1CC21 N1(C(C2CNC(=O)N2)=O)CCC2(CO)CN(C(=O)Cn3cnnc3O)CC2C1 C=CCC(F)(F)C(=O)NCC1CCCC1C(=O)N(C(C)CN(C)C(=O)NC)C C(=O)(C(C)(C)C(=O)N(C)C)NCC1(CNC(CC2(NC(C)=O)CC2)=O)CC1(F)F CC(C)C(CCNC(=O)CC1CC1(Cl)Cl)N=c1[nH]c2ccc(O)cc2s1 N1(C(C2CC(C#C)(O)C2)=O)C2CCC(C2)C1CC(=O)NCc1cn(C)nn1 N1(C(CN2CCC(NC(C3CC34CC4)=O)CC2C2CC2)=O)Cc2ccccc2C1 c1(C(c2nnnn2C2CCCC2)NC(c2sccc2Cl)C)cccc(F)n1 C(=O)(C(CNC(C1CN(C)CCO1)=O)C(C)(C)C)NCC(COCC)O c1(C(N2C(CNC(c3c(O)cccc3Cl)=O)C=CC2)=O)nnc(O)cc1O c1(C(Cc2ccc(Cl)cc2)NC(=O)CC2CCOCC2)c(Cl)cnc(F)c1Cl c1(C(N(c2c(C)ccc(Br)c2)C)=O)n[nH]c2ccc(C(F)(F)F)cc12 c1(C(=O)NCC2CN(Cc3nccc(C)n3)C2)cc(=O)c2cc(F)ccc2o1 N1(C(C(=O)NCC(CC)(N)CC)=O)CC2CCC1CC2 c1(C(C(=O)N(C)CC2(C)CCCC2)NC(CSCCC)=O)ccc(C(Cl)Cl)cc1 C1(CNC(c2ccnc(C)c2C)=O)CC12CCN(C(=O)C(C)(C)CO)CC2 C(=O)(C1CCCn2nccc21)N(CCNC(c1c(C)nn(C(C)C)c1)=O)C1CC1 CC(C)C(C)C(C)CC(=O)NCC1CN(C(=O)C(CO)c2ccccc2)C1 N1(C(C(CCCC)O)=O)CC2CCN(C(c3ccc(COC)cc3)=O)C2C1 c1(CNCc2ccc(NC(N(c3cccc(F)c3)C)=O)cc2)cc(Cl)ccc1Br c1(C(N2CC=CC(NC(=O)CCc3ccc(Cl)nc3)C2)=O)cnc2cccnn12 Cc1cccnc1CCCNC(c1ccnn1C1CCCC(C)C1)=O c1(C(N2C3(CN(C(=O)Cc4cccnc4)C3)CC2)=O)c(F)cc(Cl)cc1F CC(=O)CCCCC(=O)NC(C)(C)C(C)CC(=O)NCc1cncnc1 N1(C(c2cccc(C(C)=O)c2)=O)CC(CNC(=O)CC2OCCC2C)CC(C)C1 N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)Cc2cscn2)C(n2cccn2)C1 C1(OC)CN(C(=O)CCOCC(F)(F)F)CC1NC(c1cccn1C)=O c1(C(=O)NCc2c[nH]nc2-c2ccccc2)ccccc1OCCO N1(C(=O)OC(C)(C)C)CCC2(CCC(NC(c3nsc(C4CC4)n3)=O)OC2)CC1 c1(C(=O)N(C2CCCC2)Cc2ccccn2)cnnc2ccccc12 c1(NC(CC2(N(C(C(C)n3ccnc3)=O)C)CC2)=O)ccc(F)cc1O C(C1c2ccsc2CCN1C(=O)C(=O)NCCOC)NC(COC)=O N1(C(c2ncccn2)=O)CCC2(C1)CC2(F)F.C(CS)(CO)NC(=O)CS CCC(C(=O)N(C)CCN(C(=O)Cc1ccc(OC(F)(F)F)cc1)C)C(F)(F)F N1(C(C(C)S)=O)CC2(CO)CC1(C(N1CC(c3nccc(O)n3)C1)=O)C2 S(=O)(=O)(c1cc([N+](=O)[O-])c(Cl)cc1F)N(C1C(C)CCNCC1)C1CCSCC1 CC(C)[Si](C)(C)OCC(O)CN(C(=O)CN1CC2C=CC1C2)C C=CC1(CC(=O)NCC2(F)CCN(C(=O)C(C)CCOC)C2)CCOCC1 C#CCCC(O)C(=O)N1CCC(CNC(c2cnc(OCC(F)F)c(Cl)c2)=O)C1 C1(NC(C2C3CCCC23)=O)CCCCCC1C(=O)NCCC1(OC)CCC1 c1(C(=O)NCC2CCN(C(c3cc(OC)ns3)=O)CC2C)cccc2ncnn12 C1(C)(NC(C(C(C)C)c2ccc(F)cc2)=O)CCCN(C(c2nncn2C)=O)C1 CCCC(C(O)C(=O)N=c1ccn(CC)[nH]1)NC(=O)C(CC1CCCC1)CC N1(C(c2cc(OCC)ncc2)=O)CCN(C(C2CCCOC2)=O)CC1C CCC(O)(CC)CC.c12coc(n1)C(C)N(CC)C2=O.c1(CCC(=O)c2ccco2)cncn1C C1(CNC(c2n(CC=C)ccc2)=O)CN(C(=O)C(F)OC(F)(F)F)CCCO1 c1(C(=O)NC(CCCC)CNC(=O)CN(C)C2CC2)cc(C)ccc1O C1(C(=O)NCC2(c3ccccc3)CNC2)(CCl)CN(c2ncns2)C1 C=C=CCCC(=O)NC1CN(C(=O)Cc2cnn(C)c2C)CC1C CCC(CC(=O)NC1(CN(C)C(C2CC(n3cnnc3)C2)=O)CC1)C(C)C c1(CCC)ccc(C(C2CCN(C(=O)C(C)C(=O)O)CC2)N(C)C)cc1 c1(C(N2CC(NC(=O)C=Cc3ccco3)C(F)CC2)=O)nccc2cc[nH]c12 N1(C(c2ccc(C)cn2)=O)CCC2(CO)CN(C(=O)CCOC3CC3)CC2C1 CCC(C)(F)C(=O)N(C)CC1COCCN1C(c1cn(CCO)nc1C)=O c1(C(C(N2CC(CNC(C3(CCC)CC3)=O)C(O)C2)=O)C)cccc([N+](=O)[O-])c1 N1(C(CC2CN(C)C2)=O)CCCC2(CCC2NC(=O)CS(C)(=O)=O)C1 c1(N2CC(O)(C(C)NC(=O)CC3(C)CCCCC3)C2)ncnn2cccc12 Cc1ccnc(C(=O)NCC2CCCN(C(=O)C(c3cccnc3)C)C2)c1N C1(C(N(CCC)C(C)C)=O)CCC2C(CC1)C2(F)F.C1(=CC(=O)OC)CCOCC1 C1(C(N(C)CC2CCN(C(C(C)c3ncco3)=O)CC2)=O)Cc2nccn2C1 C1(C(N2CCN(CCN(C(C3C(C)OC(=O)N3)=O)C)CC2)=O)CN2CCN1CC2 c1(C(N2CC3CN(C(CN(CCC)C)=O)C3C2)=O)ccc2c(c1)NC(=O)C2=O CC(Cl)(Cl)C(=O)NCC1CC(CNC(=O)CC(=O)NC2CC2)CO1 C(=O)(C1CC(=O)Nc2ncccc21)NC(CNC(c1c(C)scc1)=O)(CO)CO Cc1nn(CC(=O)NC(CCNC(=O)C(C)CF)C(C)C)cc1Cl C1(C(=O)N(C2(CC#C)CCOC2)C)CCN(C(C2CC(OC)C2)=O)CC1 N1(C(c2cn(C)nc2)=O)CCCCC(CNC(=O)CC2(CO)CC2)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC(CC=C)(NC(c2ncccc2Cl)=O)C1 N1(C(c2c(CC)cccc2)=O)CCc2sccc2C1CNC(=O)CC1CCCC1 c1(N(C)CCC2CSC2)ncc(S(=O)(=O)N2CCCC(OC(F)F)C2)cc1Cl N1(C(CCC(=O)NCC)=O)CCN(C(c2cn(C(C)C)cn2)=O)C(C)CC1C Cc1cc(C)c(C(=O)NCC23CC(CN2C(C2CC(O)CN2C(N)=O)=O)C3)[nH]1 c1(C(CNC(N(C(C)Cc2cnsc2)CC)=O)C)ccccc1 C1(C(=O)NCCn2ccnc2)C2CN(C(=O)C(c3cccc(F)c3)O)CC12 c1(NCc2ncc(C)c(Br)c2)c[nH]c2cc(F)c(F)cc2c1=O c1(C(N2CCC(NC(=O)C=CC=C(Cl)Cl)(CO)C2)=O)ccc(O)c(CO)c1 c12ccc(Cl)cc1CN2C.CC(C)(Cc1cnn[nH]1)C(=O)N1CC(CO)C1 C1(C(N2CCN(C(CN(C(C(CC)CC)=O)C)=O)CC2)=O)CS(=O)(=O)CC12CC2 C1(F)(CNC(C(C=C=C)C)=O)CC2CCC(C1)N2C(c1ccc(OC)nc1C)=O c1(C(N2C(CCCNC(=O)Cc3cnsc3)CCCC2)=O)cc(O)cc(F)c1 C(=O)(CCCC(C)(C)C#N)NCC1(CNC(C2C(CC)CCC2)=O)CC(F)(F)C1 Cc1c(Br)c(C(=O)NCC2C3CC2N(C(C2(F)CC=CC2)=O)C3)nn1C N1(C(C(=O)NCC(C(C)C)c2ccnn2C)=O)CCN(c2ccccc2)C(=O)C1 N1(C(C(CC(C)C)NC(C)=O)=O)CC(C2CN(C(=O)Cc3ccns3)C2)C1 CCC(C)(C)C(=O)N1CCOC(CCNC(=O)CN2CCCCCC2)C1 C(C)(CCN=c1[nH]ccc(C#N)c1[N+](=O)[O-])NC(COc1c(C)cccc1)=O C(C(=O)NCCC1CCCN1C(=O)COc1cnn(C)c1)(C(C)(C)C)N(C)C c1(OC)cc2c(cc1F)N(C(=O)C(C)CNC(=O)OC(C)(C)C)CC2C c1(OC)c(C(=O)NC2CN(C(=O)CCCc3ccsc3)CC2C)ccnc1Cl N(C1COc2cccc(Cl)c21)C(=O)NCc1nc(C)on1 c1(C(=O)NCCC2(O)CN(C(CCCCC#C)=O)C2)ccc(N)c2ccncc12 C1(C(N2C(CCC(=O)NC(CCSC)(C)C)CCC2)=O)C(C)(C)C1(F)F C1(C(=O)NC(c2ccno2)C)CC12CCN(Cc1ccc(I)c(F)c1)CC2 c1(CC)cccc(N(C(=O)NC2CCOC2C(N2CCN(C)CC2)=O)CC)c1 c1(N(CCOC)C)ncccc1S(=O)(=O)N1CCC(CO)C(C)C1 C(CC(C(=O)NCC1CNC(=O)O1)NC(C1C=CC1C(C)=O)=O)OC c1(C(N2CCCC2CC(C)C)C(=O)NCCC)cnc(O)c(C(F)(F)F)c1 C1(NCc2c(C)nco2)CCN(C(=O)C=CCO)CC1C c1(N(C(=O)CC2(n3cnnn3)CCOCC2)C)cnc2c(c1)CCC(=O)N2 N1(C(CC(=O)NCC)=O)CC(O)CCC1C(N1CCC(C(C)O)CC1)=O c1(C(N2CCC(c3ccc(C)cc3)CC2)C(=O)NC(C)C)n[nH]c2ccncc12 C1(N(C(C(C)O)=O)Cc2ccccc2F)CCC(CNC(C2CCCS2)=O)CC1 C1(CNC(Cn2c(C(C)C)ncc2)=O)CC(NC(=O)Cc2ccon2)C1(C)C Cc1nc(Cl)sc1C(C(=O)NC1COC1)N(C1CCC1C)CC1CC1 N1(C(c2nc(CC)sc2N)=O)CC2(CNC(=O)CCC(C)OC)CCC1CC2 CC1CCCN(C(C2CCCC23CC3)=O)C1CNC(=O)CCC(C)(F)F c1(CCC)ccc(CC(=O)N(C(CNC(C2CC3CC3C2)=O)CC)CC)cc1 CC1CN(C(c2ccc(SC(F)F)cc2)=O)CCN1C(=O)CC1COCCN1C c1(-n2cc(C3N(C(c4scc(C)n4)=O)CCC3C)nn2)ccc([N+](=O)[O-])cc1Cl C12(CN(C(N3CCCC3C3CCOC3)=O)C3CC3)CCCC1CCC2 CC(C(O)C(=O)N(CC(C)(C)NC(c1ccc[nH]1)=O)C)c1ccccc1F C12(CNC(CCN(CCCO)C(c3n(C)ncc3C#N)=O)=O)CCC(CC1)C2(C)C Cn1cnn(CC(=O)NCCC2CN(C(c3cccc(Br)c3)=O)C2)c1=O c1(C2(Cn3cc(CC)nn3)CCC2)ccc(S(=O)(=O)NC2CC=CCC2C)cc1 CS(=O)c1ccccc1C(=O)NC12CC1CN(C(C1CCCCCC1)=O)C2 CCCC(C)CCNC(=O)C(C(C)O)NC(=O)CC(C)C C(C(=O)NCCNC(=O)CNC=O)OCCC.C(C)(C)(C)OC(C)=O CC(C)C(F)(F)CC(=O)NCCCCN(CCCNC(c1cnsn1)=O)C C1(CCN(C)C(C2(C)CCC2)=O)CCN(C(c2cc(C(F)F)cs2)=O)CC1 N1(C(C2=C(C)OCC2)=O)CCCC2(CC(NC(=O)CC3(C)CCCO3)C2)C1 C(=O)(C1Cc2ccc(C)cc21)NCCCCCNC(COCC(=C)C)=O N1(C(c2scc(C)c2)=O)CCC2(CCCC2C(=O)NC(c2ccno2)C)C1 c1(NC(C23CC(c4nn[nH]n4)(C2)C3)=O)cc(OC(F)(F)F)ccc1C1CC1 N1(C(C2CCN(C(=O)C3COCC(C)O3)O2)=O)Cc2cccc(C#N)c2C1 Cc1ccc(C(N2CCN(C(c3cn(C)[nH]c3=N)=O)C(CC(F)F)C2)=O)cc1Cl N1(C(=O)C=CC2CCCN2C(=O)COc2ccsn2)CC2(CCOCC2)C1 N1(C(C(CC)(C)O)=O)CCC(C2CCN(C(C3CCC=CCCC3)=O)CC2)C1 c1(C(=O)NC2CCC(C)N(C(C3CC3F)=O)C2)cc(C#N)ccc1O N1(C(C=CC(C)C)=O)CCC(C)CC1C(N1CCC(C(C)C)C1)=O c1(C(=O)NC2(C)CN(C(C(C(C)C)SC)=O)C2)cc2cccc(C)c2o1 N1(C(c2cc(C)sc2)=O)CCN(C)CC1CNC(C1CCC2CC12)=O N1(C(CC(C)C2CCCO2)=O)CCCC2CN(CCN3CCNC(=O)C3)CCC12 c1(CC(=O)NC2(C)CN(C(=O)C(O)C3CCCC3)C2)cccc(N2CCCC2)c1 C1(NC(COC2CC(NC(c3cnc(CC)o3)=O)C2)=O)CCOC1(C)C C(C)(C(C)C(=O)NCC(N)=O)NC(c1cnc(OC)s1)=O c1(NCC(CNC(c2cnc(CC)[nH]2)=O)C)nc(C(C)CC)ccc1C#N c1(C(=O)NCCNC(C2CC(F)(CO)C2)=O)cc2cccnc2[nH]1 C(=O)(C(C)CCC(=O)OC)N(C1CCN(C(=O)C(F)(F)CO)CC1)CCOC N(C1c2ccccc2CC1O)C(C1CCN(C(C2C(C(N)=O)C2)=O)C1)=O c1(C(=O)NCCN(CCC)C(c2ccc(SC)s2)=O)nc2ccccn2c1F C#CC1(OCC(=O)NCC(=O)NCCC(=O)NOC2CCCCC2)COC1.ON O=S1(=O)CCCCN1c1cccc(NC2CC3CCCC23)c1 Cc1cc(N)c(C(=O)NCCCC(CO)NC(=O)CCCn2cccn2)c(F)c1 Cc1ccc(C(=O)OCC(N2CCN(C)C(c3nccn3C)C2)=O)cc1F c1(C(=O)NC2C(NC(C(CO)NC(N)=O)=O)CC2)ccc(Cl)c(S(C)(=O)=O)c1 CCC(CC)(C(=O)NC1CC2(C1)CC(CNC(=O)CC1CCCC1O)C2)OC c1(N2C(CC(C)C)CSCC2)ncc(Br)cc1NC(=O)OC(C)(C)C C1(NC(C(CCC)CC2CCCCC2)=O)CC2CCC1N(C(=O)COCCO)C2 N1(C(C(CC)NC(C)=O)=O)CC(CC(=O)NCCCC2CCOCC2)CC1C c1(CC(=O)NC2CN(C(Cc3ccc(C)nc3)=O)C(C)C2)cccc([N+](=O)[O-])c1 C(=O)(C1=C2CCN=C2NC=C1)NC1C(CNC(COCC(C)C)=O)CCC1 C(c1csc(Br)c1)=CC(=O)OCCOC1CCCS(=O)(=O)C1 c1(N2C(C(N(C3CN(c4ccccc4)C3)C)=O)CCC2)nccc(S(C)(=O)=O)n1 C12(CC)CN(C(=O)CCCN3C(=O)CCC3=O)C(CNC(=O)C(O)C3CC3)(C1)C2 c1(CC)nc(C)sc1C(N1CC2CC2(C(N2CCC(COC)C2)=O)C1)=O N#Cc1ccnc(C(=O)NCCCOCCOCc2cccnc2)c1 CS(=O)(=O)CCC(=O)N1CC(F)(CNC(=O)CC2COCCO2)C1 CC(CCC(C)(C)C)NC(=O)C(CC1CC1)NC(=O)CC(C)c1ccco1 Cc1cccc2c1CCN2C(C1CC2C=CC1N(C(=O)C(=O)NC1CC1)C2)=O c1(N(CC=C)C(c2cnc(N3CC(C4CC4)C3)c(Cl)c2)=O)cc2nc(C)ccc2o1 c1(C(=O)NCC2CCN2C(C2CC(C3CCC3)C2)=O)ccc2c[nH]nc2c1 C=CCCCC(=O)NCC1CC1CNC(C1CCN(Cc2cccnc2)CC1)=O c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(C)[nH]2)=O)ccccc1F Cc1ccc(C(c2ccccc2)OCC(N2CCCC2c2ncc[nH]2)=O)c(C)c1 C1(NC(c2cncc(-n3ccnn3)c2)=O)C=CCN(C(C2CC2[N+](=O)[O-])=O)C1 C1(CNC(CSc2nc(C)[nH]n2)=O)CCN(C(=O)CC2CC(F)(F)C2)C1C1CC1 CCC(C)CCC(=O)N(C)CC1(O)CCCN(C(c2ccc(N(C)C)nc2)=O)C1 N1(C(C(C2CCC(=O)N2)C)=O)CCC2C(C(=O)N(C3CC(O)C3)C)C2C1 Cc1nc(N(C)C)sc1C(=O)NC1CC(C)N(C(c2cnn(C(C)(C)C)c2)=O)C1 n1(CC(=O)N(CCCC(=O)NCC2C(C)(C)C2(C)C)C)cnc2ccccc12 N1(C(C(C)NC(=O)C2CC2)=O)CCC(C(C)(O)CNC(c2cn(C)nn2)=O)CC1 c1(C(=O)NC(CCCC)CNC(=O)C=CC2CCCN2C)cc2scc(Cl)c2[nH]1 C1(C)(C=O)CCC1.N1(N(CC(=O)OC)CCOC)CCC1CO c12ccccc1NC(=O)CC2.C1(CNC(C2(SCC)CC2)=O)CC(C)(C)C1 C12(C(=O)NCC3(F)CCN(C(CC4(C)CCOC4)=O)CC3)CCCCC1OCC2 Cc1cc2[nH]c(C(N3CC4CCC4(CCNC(=O)OC(C)(C)C)C3)=O)cc2o1 C1(CC)CCCN(C(C2CCC3(CC3)C2)=O)C1CNC(=O)C(O)C(C)(C)C c1(CN(C(N(CC)CC)=O)Cc2ccccn2)cn(C)c(-c2ccccn2)n1 C1(NC(C(CSC)O)=O)CC2CCC1(C(=O)Nc1cc(F)ccc1O)C2 C(=O)(C(O)CCCc1ccccc1)NC1CC(OC)CN(C(=O)C(C)C)C1 c1(CC)nn(C)c(CC)c1CNC(C1(CS(C)(=O)=O)CC1)=O C1(CNC(c2c(SC)n(C)nc2)=O)CC(F)(F)CN1C(c1csc(O)n1)=O c1(CN2C(C(=O)NC3CCC(F)(F)C3)CSCC2)cc(O)c(O)c([N+](=O)[O-])c1 c1(NC(C2CN(c3ccccc3)C(=O)O2)=O)nc2ccccc2n1C1CC1 c1(C(C)(C)C#N)ccc(C(=O)NCC2COCCN2C(C2CCCCO2)=O)cc1 C(CCCCC(=O)NCCOC1CN(C(=O)CC2CCCN2C)C1)NC(N)=O c1(C(=O)NCC2CC(C)N(C(=O)C=Cc3ncc[nH]3)C2)c[nH]c2cccnc12 O=C(CCCCc1cnn[nH]1)NCCN(C(c1cc[nH]n1)=O)C(C12CC1C2)=O N1(C(CSCCC)=O)CCC2(CCC(NC(C34COC(CCO3)C4)=O)CC2)C1 C1(C(=O)NC(c2ccccn2)CC)C=CC(NC(c2ccnnc2)=O)C1 CCC(CCO)NC(=O)C(C1CN(C(c2ncn(CC)n2)=O)C1)OC c1(C(=O)NC2C(C)CN(C(=O)C=Cc3cccnc3)CC2)nc2cnccc2s1 CCCC(CC(C)C)C(=O)N1CCCC1CNC(C1CC(OC)CN1CC)=O C1(C(=O)NCC2NC(=O)OC2)CC2(CCN1C(C1C3CC4C(C3=O)C14)=O)CC2 Cc1ccc(C(F)(F)F)cc1C(=O)NCCNC(C1CCCC1C)=O Cc1cccc(C(=O)NC2CCC(NC(=O)C(CO)NC(N)=O)C2)c1Cl CC(C(=O)NCCCN(C)C(c1cncc2cc(F)ccc12)=O)C(C)S(C)(=O)=O CCC(C(=O)NC(C)CCN(C)C(C1(COC)CC1)=O)SC C1(C(N2CCN(C(C=C)=O)C(C)CC2)=O)Cc2cccc(C)c2O1 N1(C(C(CC)CC2CCCC2)=O)CCN(C(c2ccc(SCC)cc2)=O)CC1C C1(N(C(CC(=C)Br)=O)C)CCCN(C(=O)CC2CCCCCCC2)CC1 C(=O)(C1CCCc2nncn21)NCC(S(C)(=O)=O)CNC(C1CC2(CSC2)C1)=O N1(C(C)C)CCN(Cc2ccc(-c3ccc(N)cc3)cc2)CC1 CC(C)(CC(F)(F)F)C(=O)NCC1CC1CC(=O)NCCN=[N+]=[N-] N1(C(C2(OCC#C)CCCC2)=O)CCC(CC(c2cn(CC)nn2)C)CC1 C1(C(N2C(C)CSCC2)=O)CCN(C(c2cc(O)nc(O)n2)=O)CC1O c1(C(=O)NC2(C3N(C(C(CCC)F)=O)CCC3)CC2)ccc(C)c(C#N)c1 N1(C(CCCCOC)=O)CCOCCC1CC(=O)Nc1cnn(C)c1C#N N1(C(C(C)(C)SC)=O)CC2CCC(C1)N(C(c1coc(CO)c1)=O)C2 C1(CNC(COCCCC)=O)CCN(C(c2cnco2)=O)C12CCC2 C1(O)(CN(C(CCSCCC)=O)C)CCCN(C(=O)CCCOCCOC)C1 C1(O)(C(C)NC(c2coc(C(C)(C)C)n2)=O)CCN(C(C2(O)COC2)=O)CC1 C1(C)(NC(Cc2cc(COC)no2)=O)CCN(C(=O)C(C)N2CCC2)C1 Cc1nc2cc(CN3CC4(CC4C(=O)NCc4cccn4C)C3)ccc2s1 N1(C(c2c(C)nn(CC(F)F)c2)=O)CC2CCCC(C1)N(C(=O)C=CBr)C2 C(=O)(C(Cn1cncn1)NC(c1ccncc1)=O)NC1C(C)C1C C(C(C)(O)C(=O)N1CC2C(CNC(=O)C(F)(F)c3ccccc3)C2C1)OC c1(C(N(C)CC2N(C(C(C)OCC3CCCO3)=O)CCC2)=O)cc2c(s1)CCC2 c1(C(N(CC(N2CC(CC)(CO)C2)=O)CC#C)=O)cccc(C)n1 c1(OCC)c(Cl)nc[nH]c1=NCc1nccc(C#N)c1F C(CCCCC(=O)N1CCC(C(F)C(=O)NC2CC(CO)C2)C1)=CC C12(C(N3CC4C(NC(=O)Cc5n[nH]c(=N)s5)C4C3)=O)CCC(C(C)=O)(CC1)CC2 C1(NC(c2c(C)snn2)=O)CCN(C(=O)CCCC2CCCCC2)CC1C(C)C c1(OC)cccc(-n2cc(CNC(=O)C(C)OCCC(=O)O)nn2)c1 c1(N2CCCC(COC(C)C)C2)nc(=NCC(C)(C)CC(C)O)[nH]c2c1CSC2 N1(CCNC(C2(CNC(COCCOC)=O)CCC2)=O)CC2CC2C1 N1(C(CN(C)C2CC2)=O)CC2CC1CCN2C(c1ccc(-n2cccn2)cc1)=O N1(C(CCC(=O)NC)=O)CCCC1C1CCCN1C(=O)COCc1nc[nH]n1 C(=O)(CCC1=CCCCC1)N(C1OCC(CSC)C1)CC(=O)NC1(C)CCCO1 c1(C(=O)NC2C(NC(C(C=C)(C)CC)=O)CC2)cccc2c1CCN2 C1(NC(c2cncc(C)n2)=O)CCCCN(C(=O)CCCn2ccnc2)C1 N1(C(CC(CC)(C)C)=O)CC2CCC1C(CNC(=O)CCNS(=O)(=O)CC)C2 C1(CC(=O)NC(=O)NC)CN(C(C)(C)C)CCN1C(=O)NCC1(O)CC2CCC1C2 c1(C(N2CCC(C(C)(C)NC(COCCCCCC)=O)C2)=O)cnn(C)c1Cl c1(NC(C2C(CC)CCCN2C(C2CCCC(=O)N2)=O)=O)cn(C)c(=O)nc1O C1(C(N2CC(C=C)(O)C2)=O)CC2CCC(C1)N2C(C1CCC(C(N)=O)C1)=O C#CC1(C(=O)NCC2CCCN(C)C2)CCN(C(=O)CCc2nc[nH]n2)CC1 c1(C(N2C(=O)C2)C)ccc(F)cn1.C1(C(=O)O)CCOCC1 c1(C(N(CCNC(c2c(OCC)ccs2)=O)C(C)C)=O)ccc([N+](=O)[O-])c(C)c1 c1(NCC(N2CCC(NC(C(C)(C)N3CCCC3)=O)C2)=O)cncc([N+](=O)[O-])c1 C1(CNC(CCOCC#C)=O)CCCC(NC(c2cc(NC)n[nH]2)=O)C1 C(=O)(CC(C)CC(C)C)N1C(C)(CCC(=O)NCC(c2ccsc2)C)CCC1 C1(CC)CN(C(=O)CC2CCC3(CC3)CO2)CCC1NC(=O)C(C)=CC(C)(C)C C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCC(CNC(CCSC)=O)O c1(CC)ccc(O)c(C(N2CCC(CNC(c3ccnnc3C)=O)C2(C)C)=O)c1 C1(CCNC(=O)Cn2cc(CO)nn2)CN(C(c2cc(Cl)n[nH]2)=O)CCCO1 c1(C(=O)NC2CN(C(c3ccc(C(CC)C)cc3)=O)C2)ccc(Cl)c(N)c1 C(=O)(CCCC(C)(C)C)NCC1CCN(C(C=Cc2occ(C)n2)=O)CC1C C(c1cc2ccccc2o1)=CC(=O)NC12C(CN(c3nccc(OC)n3)C1)COC2 Cc1cccn2cc(C(N3CCC(NC(=O)C(C)(C)OC(C)C)C(O)C3)=O)cc12 C1(C(N2CCCC(CC)(NC(=O)C=CC3CCCO3)C2)=O)CCC(N=[N+]=[N-])CC1 CC(CS(C)(=O)=O)C(=O)NCC1CCCCN1C(c1ccn(C(F)F)n1)=O C1(NC(C(CC)OC)=O)CN(C(=O)CCc2cn(C)nn2)CC2(CCC2)C1 c1(OC)ccc(CNC(=O)C(c2ccco2)NC(=O)Cn2cnnc2O)nc1 CC(C)CC(C(=O)NC(C(=O)N1CCCOC(C)C1)C(C)(C)O)C(N)=O CCC(CC)C(C(=O)N(CC(C)NC(C1CC2C(C1)C2(C)C)=O)C)OC N1(C(C(C2CC2)NC(c2cc(OC)ncn2)=O)=O)CCCCC(C)(F)C1 CCCCC(=O)C(=O)N1CC2CC(NC(=O)C(C)C(F)(F)F)C1C2 CONS(=O)(=O)c1ccc(C(=O)NCC2(NC(=O)C=CC3CC3)CC2)cc1 C(=O)(CCC(=O)NC1CCCC(CN(C)C(c2c[nH]nc2OC)=O)C1)NCCC N1(C(C(C2CC(NC(CN(CC)CC)=O)C2)F)=O)CCCC2(CC1)CC2 C1(C(=O)NC2CN(C(C3CCC(C)(C)C3)=O)C(C)(C)C2)CCc2n[nH]cc2C1 c1(C(N2CCCCC2CNC(c2sc(Br)nc2Br)=O)=O)cc(O)c(Br)c(O)c1 c1(CC)cc[nH]c1C(=O)N(CCC(=O)NC1CC1)CCO.C1(C)(C)C(=O)O1 N1(C(C(CC)SC)=O)CCN(C2CN(C(c3csnc3C)=O)C2)CC1 N1(C(CCc2onc(C(C)OC)n2)=O)CCC2(CC1)CC2NC(=O)CCSC N1(C(C(C(=O)OCC)OC)=O)CC=C(C(=O)NC(C)(CO)C2CCC2)C1 CC1(C)CCCCC1C(N1CCCC1CCCNC(C1(C)CC1(F)F)=O)=O c1(C(C(=O)NC2C(C(=O)NCC(=O)NC)CCC2)O)ccc(I)cc1 c1(OC)cc(C(N(CCOCCNC(=O)CCC(=O)N(C)C)CC)=O)ccc1N C1(C(C)C)CN(C(=O)C=Cc2cscn2)CCN1C(=O)Cc1cc(O)nc(O)n1 Cc1nsc(N(C2CCCN(C(=O)CNc3ccc(Cl)cc3)C2)C)c1C#N N1(C(c2ccc(C(C)C)o2)=O)C2CCC1C(CNC(=O)Cc1n[nH]cc1Br)C2 N1(C(N)=O)CCC(C(N2CCC(CCNC(c3cccs3)=O)C2)=O)CC1 C1(CCNC(=O)CCF)CN(C(C23CCCC(CO2)C3)=O)CCS1(=O)=O N1(C(CN(C(C2(C#N)C(C)C2)=O)CCO)=O)CC2CSCC2C1 c1(NC(N2CCC(CN3CCCC3)C2)=O)csc(CO)n1 c1(C(N2CC(CCNC(COC(C)C)=O)C2)=O)cc(-c2ccn(C)c2)[nH]n1 c1(C(=O)Nc2ccc(NC(=O)C(Cl)(Cl)Cl)cc2F)cc(Cl)c(Cl)nc1Cl CCC(C)(C)CCCC(=O)N1CC(O)CCC1C(=O)NCCc1cnc(C)o1 CC1CN(C(C2CN(C(c3csc(Br)n3)=O)CCC2O)=O)CCN1C c1(N(CC(C)C)C)ccc(C(=O)OCC=CCCNC(=O)CC2(O)CCC2)cc1 Cc1nc2ncc(C(=O)NCC3COCC3NC(C3(C)CCCO3)=O)cc2o1 C(=O)(CCC(=O)c1ccccn1)N(C(C)CNC(=O)C(C)C1(O)CCC1)C Cc1cc(NC(C23CC2CCN3C(=O)C(C)CC#N)=O)cc(C)c1 CCC(C)CCCCC(=O)NC(CNC(=O)Cc1nnc(C)s1)C(C)(C)C c1(NC(CNC(C2(OC)CCCOC2)=O)C2CCC2)nc(C(C)C)cc(C)n1 c1(NC(C(N2CC(C(=O)OC)CC23CCC3)=O)=O)cc(C)c(N(C)C)cc1Cl c1(NC)cc(Cl)ccc1C(=O)NCCOC1CCN(C(=O)C#CC(C)(C)C)C1 N1(C(CS(CC)=O)=O)CCN(C(c2ccc3c[nH]nc3c2)=O)CCC1C c1(C(=O)NCC2CN(C(CCCOCCC)=O)CC2O)cn2cccc(Cl)c2n1 N1(C(C(CCC)N(C)C)=O)CCC2(COC(CNC(=O)C3=CCCCCC3)C2)C1 c1(C(=O)NC2CN(Cc3ncn(CC)c3)CC2C#N)c[nH]c2nccc-2c1 C#CCC(C)C(=O)N1CCOC(CN(C)C(c2cnn(CCN(C)C)c2)=O)C1 c1(C(N2CCC3CCC(C2)N3C(=O)C(O)C2CCC2)=O)cn2cccc(Cl)c2n1 N12CC(=O)N(C1=O)CC(=O)N(C)CC2c1ccco1.N1(CC)CCN(C)CC1 C1(CN(C2CCN(C(C3(c4ccno4)CC3)=O)C2)C)CCC2(CC2)C1 C1(F)(C(N(C)CCc2ccncc2)=O)CCCCCC1 C#CCCCC(C)C(=O)c1cccc2c(scc1)N1CC(F)CC1CN(CC)C2=O C1(C(=O)NC(COC)(C)CO)CCCN(C(=O)C(c2ccccc2)F)C1 c1(C(=O)NC(C2CCCCN2C(=O)C2=COCC2)C)ccc(C(C)S(N)(=O)=O)cc1 c1(OCCN(CCNC(COC)=O)C(c2ccns2)=O)cccc(Br)c1 c1(C(=O)NCC2CC(C)(C)CN(C(C3CC3C#N)=O)C2)c(Cl)ccc2c[nH]nc12 C1(CCCNC(CC2(C)CC2)=O)CCCCN1C(=O)CCCNS(N)(=O)=O C(=O)(C1=CCC(F)(F)CC1)N(C1CCCC(N(C)C(c2cc(=O)n(C)o2)=O)C1)C N1(C(c2cnc(OC)s2)=O)CCC(N(C)C(c2cnc(OC)nc2)=O)C(C)C1 C12(CNC(c3c(COC)onc3)=O)CCC1CN(C(c1c(F)cccc1I)=O)C2 C1(CCNC(C2(C(C)(F)F)CCC2)=O)COCCN1C(=O)CC1CC(F)(F)C1 C=CCCCCCC(=O)N1CCC(C(N2CCC3OCCC3C2)=O)(C(C)C)C1 C(=O)(C1CCc2ccc(C)cc21)NCC(C1CCCC1)NC(C1C(OC)C1)=O N1(C(c2[nH]cc(CN(C)C)c2)=O)CC2(C1)CN(C(=O)CCC1CC1(C)C)CCO2 C(=O)(C(C)CCN(C)C)N(CCC(=O)NC1(C)CC1)CCC Cc1cc(C(=O)NCC(C2CC2)NC(C2CCCN2N=O)=O)c(N)cc1F Cc1cc(F)cnc1C(=O)NC(C(=O)NCc1cnc(O)nc1O)C1CCCC1 C(=O)(CCC(C)CCCC)N1CC(C)CC(C(=O)NC(C#C)(C)C2CCCC2)C1 c1(C(=O)NCC2(CN(C(=O)CC3CC3(Cl)Cl)C)CC2)n[nH]c2c1CSCC2 c1(O)ccc(Cl)c(Cl)c1.C1(OC)CC2(C(=O)NCC(C)(NC(=O)CC3CC3)CO)CC12 C1(C(N(CCCNC(=O)COCC(F)F)C)=O)CC12CCC1(CC1)CC2 C1(NC(c2cc(OC)nn2C)=O)C2CCC(C2)C1C(=O)NC1CCCCCCC1 N1(C(COCCC)=O)CCCC(O)(CN(C(=O)C(n2cnc(C#N)n2)C)C)C1 c1(CCCNS(N)(=O)=O)cc(=NCC(O)CC2CCC2)[nH]cn1 C1(C(=O)NCCSCCC=C)C(C)CCN1C(=O)CC(C)C1CC1 c12ccc(cc1)-n1cc(nn1)C(C)(C)CC(=O)NC2.CC(F)(F)SC1CCC1 c1(Cc2noc(C)n2)ccc(Br)cc1Cl.N12CCC(CC1)C2C.c12cn(nn1)C2 C1(C(N2C(C(=O)NCC3C4CCCOC34)CC(C)C2)=O)C2C3CCC(C3)C12 c1(CN2C(c3cccc(C)c3)C(C)CCC2)cccc2c1OCC2 c1(C(=O)NC(CC(=O)N(CCCO)CC)C(F)F)ccnc2cc[nH]c12 C1(SCC(N2CC(NC(C3CSCCS3)=O)(CO)C2)=O)CCS(=O)(=O)C1 c1(C(c2nnnn2C(C)(C)C)NCCN2C(C)CCCC2)cc(Cl)c(Cl)c(Cl)c1 c1(SCC)ccc(CC(N2CC(CCNC(c3nocc3Cl)=O)C(C)C2)=O)cc1 C12(C(=O)NC(C(C)C)CCNC(=O)C=C3CCOCC3)CCN(C1)S(=O)(=O)C2 C(=O)(C1=NN2CCCN=C2N1)Nc1cccc(CNC(CCC)=O)c1 C(CCCCC(=O)NC1CCC(CC(=O)NCCC2CCSC2)CC1)SC c1(C(C)=O)cn(C)nc1C(=O)NC1(CNC(c2[nH]nnc2C2CC2)=O)CCC1 c1(CC)nc(C(=O)NC(C)(CNC(c2ccncc2F)=O)CO)c(C)o1 c1(C(=O)NCC)ccc(OC)c(OC)c1CNC(=O)C(=O)NC1(O)CCCC1 N1(C(c2c(CC)cno2)=O)CCC(CNC(C2CCOC2(C)C)=O)CC1 CC1CCCC(CCNC(=O)NCC(c2ccccc2F)N2CCCC2)C1 C(=O)(C1=NOC(CNC(=O)CCC(C)C)C1)NC(c1ccc(C)cc1)C S(=O)(=O)(c1ccc([N+](=O)[O-])cc1)NCC(C)(C)C(=O)N1CC(CCO)(COC)C1 N1(C(c2cc(C#N)c(F)cc2)=O)CC2(C1)CN(C(C1C3CCCC13)=O)CC2CO C1(NC(c2c(C)nc(C(C)C)o2)=O)CCCC12CN(C(C1CCNC1=O)=O)C2 c1(C(N2CC(NC(=O)CC34CCC3C4)C2)=O)ccc(NS(=O)(=O)C2CC2)cc1 N1(C(CCCCC(CC)C)=O)CC23CCCC2(CN(C(=O)Cc2ccsc2)C3)C1 C1(CNC(C(C)=C2CCC2)=O)CC2(CCC2)CN1C(=O)CC1(C)CC1 C(C(CC(C)C)C(=O)NC1CN(C(c2ccc(C#N)cc2F)=O)CCC1F)OC C(N=c1nc(Cl)[nH]c(C)c1C#N)C1CCN(C(CC(C(F)(F)F)NC(C)=O)=O)C1 CC(C(=O)N1CCCC1CCC(N1CCCC(O)C1)=O)C(F)F C1(CC(=O)NC(C)(C)CCNC(=O)Cc2ccsc2)CC2CCC1C2 N1(C(c2ccc3sncc3c2)=O)CCCC1C1CCCN1C(c1ccc[nH]1)=O C1(NC(CNC(CC)=O)=O)CCN(C(=O)CCCc2ccc(C#N)cc2)CC1C C(=O)(C1=CCCCCC1)NC1C2CN(C(C(C)Cc3cccnc3)=O)C1C2 c1(OC)ccc2c(c1)CC(C(=O)NC1CCC(N(C(=O)C3=CCCC3)C)CC1)O2 C(CC)(C(=O)NCC=CCNC(=O)CCc1nccn1C)OCC C(CC(C)(C)C(=O)N1CCC(CNC(c2ccc(O)cc2C)=O)C(C)C1)OC c1(C(=O)NCCCN(C(C)C)C(C2CC3CC3C2)=O)ccc2nc(CO)[nH]c2c1 N1(C(Cn2c(C)ccn2)=O)CC(NC(=O)CO)CC(C)C1 N1(C(c2ccc(CC)cc2C)=O)CC(C2CCN(C(=O)C=Cc3ccsc3)CC2)C1 c1(C2(O)CC(C(N3CC(N(C(C4N(CC)CC4)=O)C)C3)=O)C2)ccc(F)cc1 C1(O)(C(C(=O)N(CC)Cn2ccnc2)F)CN(C(c2ccoc2C2CC2)=O)C1 C1(NC(C2CN(C(C)C)C2)=O)CC(NC(=O)CSc2cc(C)oc2C)C(O)C1 C1(NC(CC(C)OC)=O)CC2(C1)CN(C(c1cc(O)cc(O)n1)=O)C2 S(=O)(=O)(c1ccccc1F)NCCC(=O)NC12CC(CNC(C(C)C#N)=O)(C1)C2 C(=O)(C#CC1CC(F)(F)C1)NC1CCN(C(c2c(F)ccc(C)c2)=O)CC1 C1(CNC(CC2(CC)CC2)=O)CC2(CCN(C(=O)CSCCC#N)CC2)CO1 N1(C(C(COC)C)=O)CCC(CC(=O)Nc2cccc(F)c2F)C1(C)C C1(C(=O)NCCC2(OC)CN(C(c3cc(C(F)F)no3)=O)C2)CCCC12CC2 CCC(CNC(=O)CC=CCNC(C12CCC(CC1)C2)=O)C(C)C CN1CCN(C(c2ccc(C(N3CCCC(COC)C3)=O)cn2)=O)CC1=O c1(NC(NNC(c2cnc(O)cc2O)=O)=O)ccc(Br)c(N2CCOCC2)n1 c1(C(N(CCC(C)C)C(c2noc(C3CC3)n2)C)=O)nc(Cl)cc(N)c1Cl C12(CNC(C3C(C(C)C)CCO3)=O)CCC1CN(C(=O)C(C)S(C)(=O)=O)C2 CCCC(C)CC(C(=O)NC)N1CCOCC(N2CCOCC2)C1 N#CC1(N(CCN2CC3C(C2)C3(F)F)C(C2C3CC4C(C3)C24)=O)CCCOC1 N(C(=NCc1ccnn1C)NCC1CC12CC2)C(CC)CO CC1CN(C(C2CC2c2ccccc2F)=O)CCN1C(C1CCC(=O)N1)=O N1(C(C(CC(C)C)(F)F)=O)CCC2(CCC2CNC(=O)C2=CCCSC2)CC1 N1(C(C=CCC)=O)CCC2CN(C(=O)C(C3CCCCC3)CC)C2C1 c1(CN(C(c2cn(-c3ccccc3)nn2)C)C)cc2c(cc1F)NC(=O)CO2 N1(C(=O)Nc2ccc(-c3c(C)cccc3)s2)CC2CN(C)CC2(C)C1 c1(C(N(C2CCCN(C(C3CCS(=O)CC3)=O)C2)CC)=O)ccncc1C(F)F N1(C(COCC)=O)CCCCCC1CNC(c1oc(-c2cnn(C)c2)nc1C)=O CCC1=C(C(=O)NC2CN(C(=O)C(C)Oc3cccnc3)CC2(C)C)CCCO1 c1(CC(=O)NC(c2ccccc2)CNC(C2(Cl)C(C(C)=O)C2)=O)cnnc(O)c1 N1(C(C(C)Sc2ncccn2)=O)CC(NC(C2CC(F)(F)C2)=O)C(CC2CC2)C1 CCC(O)C(C)(C)C(=O)NCC1CN(C(=O)Cn2ccc(C)n2)CCO1 C1(C(=O)NCC(C)(O)CSC)CC(=O)CN1C(c1ccc(COC)o1)=O N1(C(C2(C)CCN(C)CC2)=O)CC2CCC(CNC(C3(C(C)(F)F)CC3)=O)(C2)C1 N1(C(C(CCSC)OC)=O)CCCN(C(c2ccsc2)=O)CC1C(C)C C#CCC(O)C(=O)NC(C1CCN(C(=O)CN(S(C)(=O)=O)C)CC1)C C1(C(=O)NCCNC(c2c(C)nns2)=O)CC2(CCCCC2)C1 C1(N(C(Cn2cc(COC(C)OCC)nn2)=O)C)CS(=O)(=O)CC1O C(=O)(C(CO)NC(C1(NC(=O)CC2(OC)CCC2)CC1(C)C)=O)OC C1(N(C(c2cnc(CC3CC3)o2)=O)CC2CCCN2C(C2CC2F)=O)CCC(O)CC1 Cc1cccc(CNC(C2(NC(c3cnc(N(C)C)s3)=O)CCN(C)C2)=O)c1F C(=O)(C1SCc2cccnc21)NCC(CNC(C=NOC)=O)F c1(C(=O)NCC(CC)(CC)NC(=O)C#CC2CC2)ccc(CO)cc1F Cc1cc(C(N2CCN(C(=O)CC3(O)CCCOC3)C(C)C2)=O)cn(C)c1=O N1(C(CC=CCC)=O)CC(O)CC1C(=O)NC1CC1(F)F C=CC(CC)CC(=O)N1CCC1C(=O)N(C)CCNC(C)=O Cc1nc(C2CC2)sc1C(=O)NCCC(C(C)C)NC(=O)Cn1cnc(C#N)n1 N1(C(C2C(C(C)(C)C)C2)=O)CCC(C(CO)NC(C2CCS2(=O)=O)=O)CC1 c1(C(N2CCC(N(C(C3CC3c3cncn3C)=O)CC)C2)=O)cc(C)ccc1O N1(CC(C)SC)CCN(C2CCCN(C(=O)Cn3nnnc3C)C2)C(=O)C1 c1(C(N2CC3CN(C(CS(C)(=O)=O)=O)CC3C2)=O)cncc2ccccc12 c1(CC(=O)NCC(C)N(C)C(c2ccc(C(F)(F)F)o2)=O)ncsc1Cl C1(CC(=O)OCC)CC=CCC1SC.C1(C(F)(F)F)(C(=O)OCC)CC1 c1(C(N2CCCC(N(C(C(n3c(C)ncc3)C)=O)C)C2)=O)cccc2c[nH]nc12 c1(C(=O)NC2C(NC(C3(C)CCNC(=O)C3)=O)C2)cc(N)c(F)c(F)c1Cl C1(NC(C2N(C(C3(C)N(C)CCC3)=O)CCC2)=O)CCCCCC1O Cc1c(NCC2CN(C(C)C)C2)ncnc1N1CCOC(C2CC2)C1 c1(C(N(C2CCN(C(C(CC=C)C(C)C)=O)C2)C)=O)cccc2c1CC(C)(C)C2 C#Cc1ccc(C(N2CCC(NC(C3C(C)C3C)=O)C2)=O)c(C(F)(F)F)c1 N#CC1(C(=O)NCCC2CCCCN2C(c2cc(F)n[nH]2)=O)CCCCC1 CC1(C)CN(C(=O)Cc2ccc(Cl)s2)CC(CNC(c2cc(O)ncn2)=O)O1 c1(OC)c(C(=O)NC2CC(O)CN(C(C3CCS(=O)(=O)CC3)=O)C2)cccc1Cl C(=O)(C(C)CC(=O)N1CCC(CNC(c2cc(F)ccc2C2CC2)=O)CC1)OC C1(NC(C2C(C(C)C)N(C(c3cc(C#N)c[nH]3)=O)CC2)=O)COCCC1(F)F N1(C(C=C(C)C(C)C)=O)CC(NC(=O)C=CCF)CC12CCCOC2 C1(C(C)OC)CC(=O)NCC2(CC=CC2)C(=O)N1.c1(C(C)SC)c(C)n[nH]c1C Cc1nc2cccc(Cl)c2cc1C(=O)NCCC1CCN(C(=O)CCC(F)F)C1 CC1CN(C(=O)C=CC(c2ccccc2)=O)CCN1Cc1ccc(F)nc1F C1(CC(=O)OC)CC(NC(=O)NCC(C)(C)C2CCC2)CCO1 CCCCC(F)C(=O)N1CCC(C(=O)N(CCCC)CCO)C(O)C1 c1(CCC(=O)NCC2C(NC(CC3(C)CCC3)=O)C2)cnc2n1CCOC2 Nc1ccc2c(c1)N(CC(=O)CC1COCCO1)CCC2 C(CCC1CC1)(C(=O)NC1CCOCC1)NC(c1ccn(C(C)C)n1)=O N1(C(C(CO)N(C)C)=O)CCN(C(C2CCC(C)(C)CO2)=O)CC1CO Cc1cccc(COCC(=O)NC(C)(CNC(=O)CSC2CC2)C2CC2)c1 C(=O)(CC(C)(F)F)NCC1C(NC(CC(=C)Br)=O)C1 Cc1cc(C(=O)NC(CC(=O)NC(CO)CCC2CC2)C2CC2)ns1 N1(C(C2(CNC(C3C(COC)CC3)=O)CCCO2)=O)CC2(C1)CN(C)C2 c1(CSCC(=O)NC(C2CCN(C(c3ccncc3)=O)CC2)C)ccccc1Cl CC1CN2CC1CC1(CC1)C2=O.C(=O)(CCc1cccs1)NCC1CCC1 C1(N(C(C(c2ccccc2)C)=O)C)CN(C(=O)CCC#N)CC1(C)C N1(C(C(C2CCCN(C(c3cnsc3)=O)C2)C)=O)CCN(C)CC(O)C1 CN1C(=O)CCCC1C(=O)NCC1C=CCN1C(c1cc(C2CCCC2)[nH]n1)=O N1(C(C2C(C)CCO2)=O)CCC(F)(CNC(=O)CN(C)C(N)=O)C1 c1(OC)cccc2c1C(C(=O)NCC1(NC(=O)C3=CCCS3)CCOC1)CC2 n1(CCC)cncc1CNC(=O)CSCCNC(=O)CC1CC=CCC1 C1(NC(c2nn(CC)c(O)c2)=O)CN(C(=O)CCc2cnc[nH]2)CC12CCCC2 c1(SCC)cc(C(=O)NC2CC2NC(=O)Cc2nc(CC)no2)ccn1 Cc1cc(C(N2CCOCC2CNC(c2ccnnc2S)=O)=O)cc(O)c1 C1(NC(C2CCC(C)O2)=O)CN(C(=O)Cc2cnccn2)CC2(CC2)C1 C1(C#N)(C(=O)NC2CCC(N(C(=O)C=Cc3ccncc3)C)CC2)CC2CC2C1 c1(C(=O)NCCN(C(C(COC)C)=O)C)cccc(N2CCCC2=O)c1 CC(C)C(C(=O)N1CCCC(Cn2cc(CO)nn2)C1)N1CCCC1=O S(=O)(=O)(CCC(=O)NCC1CC(NC(C2CC=CCC2)=O)C1)N(C)C c1(OC)ccc(CC(=O)Nc2ccc(NC(c3cocn3)=O)c(C)c2)c(F)c1 CCCCC(C(=O)NCC1=CCN(C(=O)CCc2cncnc2)CC1)C(C)C N1(CC(=O)NC(CC(C)NC(c2c[nH]nc2F)=O)C)CCCCCC1=O CC1(CNC(=O)C(CC2CC2)NC(=O)CN2CCCCC2)CC2(CC2)C1 C1(C(N(CCCCOC)C)=O)CC2CCC(C1)N2C(=O)Cc1nonc1C c1(C(=O)NCC2(CNC(C3C(OC)CCCC3)=O)CC2)cnn2ccsc12 C(=O)(CCS(N)(=O)=O)NC1CCC(CC(=O)N(C)CCOC2CC2)CC1 C1(CC(N2CC(CN(C(C(C)C#N)=O)C)OCC2)=O)CC2CCC1CC2 N1(CC)CCc2ccc(NC(c3cc(C(F)(F)F)nn3C)=O)cc2C1 C(=O)(CC(C)(C)c1ccccc1)N(C1CN(C(=O)Cn2cc(Cl)cn2)CC1F)C c1(C(=O)NC2(C)CCCN(C(=O)CN3CSCC3=O)C2)cnc2nccnc2c1 c1(C(N2CCC(NC(C3CC(C)OC(C)C3)=O)CC2)=O)cc(Cl)cc(Cl)c1N C(=O)(C1=CC(C)(CC(=O)OC)C1)NC(C1CCCCC1)CNC(CCC#C)=O N(C(=NCCF)NCC(c1ncn(C)n1)(C)C)C(c1ccccc1Br)C C(=O)(C1=Cc2cccc(Br)c2OC1)NCCNC(c1c(C)ccc(O)c1)=O Cn1nccc(C(=O)NCC2(C)CCN(C(C3CC(=C4CC4)C3)=O)CC2)c1=O N1(CCCC)CC(C(=O)NCCOCCOCCNC(=O)CC)CC1=O CCCC(O)C(=O)N1CC(CC(=O)NC2CCCN2C=O)(OC)C1 CC1C(c2ccccc2)CCN1C(=O)CCc1ccnn1C N(C(=NCCCN1CCOCC1)NCCC1CC(OC)C1)CC1(OCC)CCC1 Cc1ccc2c(c1)CC(C(N1CCN(c3snc(C)c3C#N)CC(O)C1)=O)S2 c1(C(=O)NC2C(C)CN(C(=O)CCC(C)(F)F)CC2)cnc2c(=O)[nH]ccc2c1 Cc1nccc(C(=O)N(C2CCN(Cc3cc(Br)co3)C2)C)n1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)NCC1N(C(C(CCC)OC)=O)CC(F)C1 C1(NC(CCOCC)=O)CC2CN(C(=O)CN3CC(C)C3)CCN2C1=O c1(Cc2cc(C)n(C)n2)cc2ccccc2o1.C1(NC(=O)N)(C)CCCCC1 N1(C(C2(C(=O)O)C(c3ccc(C)cc3C)C2)=O)CCC(O)C12CCCCCC2 C1(CNC(C(C)COc2ccccc2)=O)(NC(C2CC2F)=O)CC2CCC1CC2 c1(CC)ccc(C(=O)NC2(CO)CCCN(C(C3CC4(C3)CC4F)=O)C2)c(O)c1 Cn1cc2ccc(C(=O)NCC3CN(Cc4ccc(O)c(Cl)c4)CCO3)cc2n1 N(C(=NCC(C)C)NC(c1ccccc1C)C1CCOC1)C1CC(OCC)C1 N1(C(CC(COC)C)=O)CCC(C)CC1C(=O)N(C(CF)CF)C C12(CNC(c3c(CC)ncs3)=O)CC(CNC(=O)C(C)OC)(CO1)C2 c1(CC(N2CCN(C(C3CC(C)C3)=O)CC2CC(F)F)=O)ccc2nonc2c1 C(=O)(C(C)C(C)S(C)(=O)=O)NCC1OCC2(CN(C(c3cn(CC)nc3)=O)C2)C1 c1(C(N(S(=O)(=O)C2CCCCC2)C2(CN)COC2)=O)ccc2ccncc2c1 c1(OC)ccccc1CN(C(=O)CN1CC2CCC1C2)C(C1OCC1(C)C)=O N1(CCN(C(=O)CC=CCNC(C2CC2C2CCCO2)=O)C)CCCCC1 C12(C(=O)NCC=CCNC(C(C(C)O)N(C)C)=O)CCC(CO)(CC1)CC2 C1(C(=O)NC(CC)(CNC(=O)CCC2CCC(C)O2)CC)CC2CCC1CC2 Cc1ccc(CNC(C2CCC(CNC3CCC=CCC3)C2)=O)nc1 C1(C(=O)NCCN(C(C2(CC=C)CCC2)=O)C2CC2)CCCCC1(C)C c1(C(N)=O)cc(NC(=O)NC2CC2CNC2(C(F)(F)F)CC2)ccc1F C=CCC(C(=O)NCC1CN(C(=O)C(C2CCC2)OCC)CC(C)(C)C1)C(C)C N1(C(CSCCOC)=O)CCC(C2CC2)C1CNC(=O)CCc1nnc(C)n1C CN1CCCC(F)(C(N2CCCC(CNC(C3(C(=O)C4CC4)CC3)=O)C2)=O)C1 C1(CNC(=O)C=CC2CCOCC2)CCCN(C(c2cc(O)no2)=O)CC1 N1(C(C2CC23CCCC3)=O)CCC2(CC1)CC2C(N1CCC2CC12)=O C(=O)(CC(C)(C)C(C)=O)N(CC(=O)NC1CCOC1C)CC C1(CC(=O)NC2CC(C(C)NC=O)C2)CC2CCC1CC2.c1cncc(C#N)c1 N1(C(C(=O)Nc2c(C)c(Cl)ccc2)=O)CC2C=CCOC2C1 CN1CCC(=CC(=O)N(CCNC(C2(C)CC2F)=O)CC2CC2)C1 c1(CC)cc(C)ccc1NC(=O)CCC1CC(NC(C2CC=C(C)CC2)=O)C1 C1(C(N(CCNC(c2cncc(C)c2)=O)C2CC2)=O)CCn2cc(C)nc2C1 C1(NC(=O)C2=CCCS2)CCCCCN(C(c2cc(C(F)F)ccc2F)=O)C1 C1(C2CCN(C(=O)Cc3nnn(C(C)(C)C)n3)CC2)(NC(CCC2(C)CC2)=O)CC1 c1(OC)nccc(=NC2CC2c2cccc(C(F)(F)F)c2)[nH]1 C1(C(N2CC(=C(CNC(c3c(Cl)nsc3Cl)=O)F)C2)=O)Cc2ccncc2C1 C(=O)(CCCC(=O)Nc1cccc(CNC(=O)Nc2cc(Cl)ncc2C)c1)OC c1(CN)ccc(Cl)c(O)c1.n12nccc1C(=O)N1CC(C1)NC(=O)C21CC1 c1(C(c2ccccn2)SC(C)C(=O)Nc2ncc[nH]2)ccc(F)cc1 C1(NC(c2cnn(C)n2)=O)CCC2(CC1)CN(C(C1C3CCCC13)=O)C2 c1(OC(C)C(=O)NCC2(F)CCN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)ccccc1F C(CC(C(=O)NCC1(CO)CCOC1)NC(c1cc(C)sc1C)=O)=CC c1(C(=O)NC2CCC(CCC(=O)N(C)Cc3ncn(C)n3)C2)cccn2ccnc12 C1(OCC(NOC2CCN(C(CCOC)=O)CC2)=O)CC2CC1CC2O CCC(CC)CCC(=O)NCCc1n[nH]cc1C(=O)NCC1CCOC1C(C)C C(=O)(CCCCCC(C)C)N1CC(O)(C(CNC(C(CC)OCC)=O)(C)C)C1 Cc1nnc2n1CC(C(N1CC(CNC(=O)CC(F)F)CCC1C)=O)CC2 c12ccc(cc1)OC(=O)C2.c1(NC(N(C)C(N)=O)=O)cc(-c2ccco2)on1 Cn1cc([N+](=O)[O-])cc1C(N1CCN(C(=O)C=CC(c2cnn(C)c2)=O)CC1)=O CN1C(=O)c2ccccc2C1CC(=O)NCC12CCC(C1)N(C(C1CC1F)=O)C2 N1(C(C(C)SCC)=O)CC2(C1)SCCC2NC(=O)Cc1cccc(Cl)c1F c1(-c2c(C)cccc2)occ(C(F)(F)F)c1C(=O)NC1CC(C)N(C(=O)C2CC2)C1 c1(CN(C2CCN(C(c3ccc(N(C)C)s3)=O)C2)CCO)cc2ccccc2cn1 c1(OC)ncc(-c2nc(COc3nccn3-c3cc(C)cc(C)n3)cs2)cc1C CC(C)C(C)CC(=O)NCC1CN(C(=O)CC2CC(C)OC2C)CCCO1 CC1(CNC(=O)Nc2ccc(C3CCC(=O)N3)cc2)COc2ccccc21 C1(N(C(=O)CC2(C)CC2)C)CN(C(c2ccnc(O)c2F)=O)CC1(C)C CC(C)(C)CC1CC1C(=O)NCCNC(C1CC1Cl)=O N1(C(=O)CC2(F)CCC2)CCC(F)(CNC(=O)COCc2ccccc2Cl)C1 C1(NC(C(C)C(C)(C)C)=O)CN(C(C2CC(C(C)C)=NO2)=O)CC2(CCC2)C1 N1(C(COCC#C)=O)CC(C)N(C(=O)CCCN2C(=O)CNC2=O)CC1C C(=O)(C(O)Cc1[nH]cnc1C)NC(CCNC(C(C)=C(CC)C)=O)C C(CC(C)(C)C(=O)NOC1CC2CCC1C2)NC(CCC1CCC(C)O1)=O c1(C(=O)NCC2(O)CN(C(C3C(C(C)C)(CC)C3)=O)C2)ccc2c(c1)CC(C)O2 C1(C(C(=O)NC(C)C)N(CC(C)OC)C)CCC2CC1C2(C)C c1(N(C2CCCN(C(C3CCC(F)C3)=O)C2)C)ncnn2c(Br)ccc12 CC(C)CCCCC(=O)NCC(CC(C)C)NC(C1CCN(C2COC2)C1)=O c1(N(C)CC2CCCCC2)cccc(S(=O)(=O)NCc2ccc(C#N)cc2)n1 CC(CCC(C)(C)C)C(=O)NC1(C)CN(C(=O)Cn2ncc3ncccc23)C1 CCCCC(CC)C(=O)NCC(C)CNC(c1c(C)noc1CC)=O CC1CCC(CC(N2CC(CN(C(=O)COC(C)(C)C(F)(F)F)C)C2)=O)CC1 C1(NC(C(C)SC)=O)CCN(C(c2ccn3ccnc3c2)=O)CC(O)C1 N1(C(CC=C(C)C)=O)CC(C(N2CC(O)(C(F)F)C2)=O)C(C2CC2)C1 c1(OC)ccc(COCC(=O)NCCCCNC(C2(O)CC2)=O)cc1OC c1(OC)ccc(S(=O)(=O)NC(C)CC(=O)NCCCCC(C)(F)F)cc1 C(=O)(C1CCc2ccc(Cl)nc21)NC1CN(C(C2(CC(=O)OC)CC2)=O)CC1O c12cccc(c1)NC(=O)NC2.c1(CC)csc(CC(=O)OCCO)n1.C1C(=O)N1 C1(CNC(C(C)C)=O)CN(C(c2cc(-c3ccccn3)ns2)=O)CCN1C CN1CCC(O)(CNC(C2(CNC(=O)C=C3CCC3)CCCO2)=O)C1 c1(C(C(=O)NCCOC)N(C)Cc2ccccc2O)cc(Cl)c2ccncc2n1 C1(C(=O)NCC2(F)CN(C(Cc3c(C)scc3)=O)C2)CCC2(CCCCC2)C1 Cc1cn2cc(C(=O)NCC3CCCN(C(c4ccc(CO)s4)=O)C3)ccc2n1 N1(C(CNC(CC)=O)=O)CC(CNC(c2n[nH]cc2C)=O)CC(C)C1 N1(C(C2(c3ccn(C)n3)CC2)=O)CCC(CNCCC2(C(F)F)CC(O)C2)CC1 N1(C(CC2CCC(=O)N2)=O)CCC2(CC(NC(=O)C=CCNC)C2)C1 C#CC1CN(C(=O)CC(C)CCC=C(C)C(c2ccc(Cl)cc2)=O)CCN1C C12(NC(CCc3ccnc(C)n3)=O)CCC(C1)N(C(=O)CN(C)C(N)=O)C2 C1(NC(=O)C=Cc2ccccc2F)CC2CN(C(c3ccc(F)cn3)=O)CC2C1 c1(C(N2CC3C(CNC(C=C4CCC(C)C4)=O)C3C2)=O)cc2c(s1)CCCCC2 c1(C(=O)NCCOC2CN(C(COCCC)=O)C2)[nH]c2ccc(F)cc2c1Cl c1(C(N2CC(OCCNC(C3CC3C3CCCO3)=O)C2)=O)ccnnc1 C1(CNC(CC(C2CC2)NC(C)=O)=O)CCCCCN1C(c1ccc[nH]1)=O C(C(O)C(F)(F)F)NC(C(=O)N(C)C(c1n(C(C)C)cnc1)c1ccccc1)=O CCCCCCCCCCS(=O)(=O)N1CCC2C1CCCN2C(=O)C(C)S CC1=CC(C)CN(C(=O)C(=O)NC2CC(C)(C)CN2Cc2ccccc2)C1 C(=O)(C1=CCCCC1)N1C(C(=O)NC2CC(C)SCC2)CSCC1 N1(C(c2cncc(C#C)c2)=O)CCN(C(C2(CF)CC2(F)F)=O)C2(CCC2)C1 c1(C(=O)NC2(c3onc(C)n3)CCC2)cc(Cl)c(S(N)(=O)=O)c(Br)c1 N1(C(C(C)=CC=C)=O)CCC(CC=C)(C(=O)NC(c2nc(C)no2)C)C1 CCCCCCC(C)(CC)C(=O)NC(C)CNC(c1cc(C)ccc1F)=O C1(C(=O)NC(CC2CN(C(C3(OCC)CCC3)=O)C2)C)CCC(OC)C1 Cc1nccc(-n2cc(C3(c4ccccc4)CC3)nn2)n1.CO C1(C(N2C(C3CC3)C(=O)NCC2)=O)CCCCCC1.c1(SC)coc(C2CC2)n1 N1(C(CN(c2cccs2)C)C)CCC(=O)N(CCN(CCCC)CC)C1=O C=C1CC2(C1)CN(C(C1N(C(C3CC(O)C(F)C3)=O)CCC1(C)C)=O)C2 Cc1cccc(C(N2CC(NCc3cccc4c3CCC4)C(O)C2)=O)c1[N+](=O)[O-] c1(NC)cccc(C(=O)NC2CC(C)(NC(=O)CCc3nc(N(C)C)no3)C2)n1 N1(C(CC(C=C)C)=O)CCC(C)(C)C1C(=O)NCC1CCCN(C)C1=O C1(c2onc(C(C)(C)OCC)n2)CCN(c2nccnc2OC)CC1 C1(C(=O)NC(c2nc[nH]n2)C)(SC)CN(C(C2CC2(C)C(F)F)=O)C1 C1(CC(=O)NC(COC)(C)C)CC2(CC2)CN1C(C1CCOCC1(C)C)=O c1(C(=O)NCC(C)(C)NC(C(CC)NC(C)=O)=O)cc(Cl)c(OC)c(Cl)n1 c1(CNc2c(C(N3CC(F)CC3)=O)nccc2)ccccc1[N+](=O)[O-] c1(C(=O)NCC(CO)NC(c2cc(C(C)C)nn2C)=O)ccc2c(c1)CC(=O)N2 n1(CCC)ncnc1C1(O)CN(C(=O)NCc2nc(C3CC3)n[nH]2)C1 C1(CNC(c2c(-c3onc(C4C(C)CCC4)n3)nccn2)=O)CC2(CC2)CN1C C(=O)(C1=NN2CCCN=C2N1)NCC(CC)NC(=O)CC(C)C(C)C C1(C(=O)NCCN(C(=O)C(c2ccnn2C)O)C)CCCN(S(N)(=O)=O)C1 C1(F)(C(=O)NC2CC3(CN(C(c4cc(C)c(C)s4)=O)C3)C2)CC12CCCCC2 c1(CC)nc(C2CCCN2C(=O)Cc2ccn(C)n2)no1 N1(C(c2onc(C)c2C)=O)CCCN(C(=O)C(C)Cn2ccnc2)CC1C c1(N2C(C(C(=O)NCC(=O)OC)(C)C)CCC2)ccnnc1Cl C1(CNC(c2csc(Cl)c2)=O)(NC(C2CCC3CCC23)=O)CCCCC1 c1(CCOC(C2C(CC)CCCC2)=O)c(C)nn(C)c1C N12CCOC(C1)C2.c1(C(N(C(C)C(C)C)CCC)=O)ccccc1Cl S(=O)(=O)(C1CCN(c2ccc(I)c(Cl)n2)C1)NCCNC C1(CNC(c2ccc(C(C)=O)o2)=O)CC(NC(c2ncoc2C)=O)C1(C)C c1(CNC(C2N(C(C3C(OC(C)(C)C)C3)=O)CCC2)=O)cnc(O)c(F)c1 C1(CNC(c2c(C(C)=O)coc2)=O)CCCN(C(=O)C(c2cnn(C)c2)O)CC1 n1(CC)cc(CNC(c2csc(Cl)c2)=O)cn1.C12CCC(O1)CN(C1CC1)C2=O N1(C(C2(CC(C)C)COC2)=O)CC(NC(=O)CN2CCC(C)CC2)C(C)C1 C(=O)(CCC1=CCc2ccccc21)NCCCC1(NC(CC2CN(C)C2)=O)CC1 c1(NC2CC3(CC(CSC)C3)C2)nc(Sc2c(F)ccc(Br)c2Cl)ncc1C#N C=C(Cl)CC(C(=O)NCC1(C)COCCO1)NC(C1CC(=O)CCO1)=O c1(C(N(C(C)CNC(=O)CCCN(C)C)CC)=O)cccc2oc(C)nc12 C1(CC(N2C3CN(C(c4c(OC)cccn4)=O)CC2C3)=O)CCn2cncc2C1 C1(C)(C(=O)NC(CCOC)CNC(c2ccc(F)s2)=O)CCC(C)CC1 CC(C)C(C(=O)NCC1CC(OCC(=O)NC(C)CCC2CC2)C1)C1CC1 Cc1scc(C(N2CCOC(C(C)NC(=O)C=C3CCSCC3)C2)=O)c1N c1(CN2CCC(C(=O)Nc3nc(C)c(Cl)nc3)C2)ccc2c(c1)CNC2=O CCC(C)C(CC(=O)N(C)Cc1ncco1)NC(C1(C)CCCC1O)=O C1(C(=O)NC2CCCCN(C(c3c(C)noc3N)=O)C2)CCCCC1C1CC1 C1(CNC(C2C(C(C)O)C(=O)C2)=O)CC(OC)CN1C(=O)CC1(CO)CC1 N1(C(C=C(C)C(F)F)=O)CCC2(NC(c3coc(-c4ccccc4)n3)=O)CC2C1 C=CCCC(C(=O)NC(c1ncn(C)n1)C)NC(c1sc(F)cc1C)=O C(=O)(CCC(=O)NN(C)C)NCC1N(C(C(C)=C(CC)C)=O)CCCCC1 CCC(CC(=O)NCC1(O)CCN(C(=O)C(C)NC(=O)CC(C)(C)C)C1)C1CC1 C1(NC(C=CSC)=O)CCC(C)N(C(=O)CCc2ccc(Cl)c(Cl)c2)C1 C12CCN(CC1O)C(=O)Nc1ccc(cc1)NC2=O.c1(NC(N)=O)ccncn1 Cn1cc(C2CCCN2c2nc(C3CCCCC3)ns2)cn1 c1(C(=O)NC2CC3(CC(NC(CCN(C)C)=O)C3)C2)ccc(Cl)c2ccccc12 c1(C(N2C(Cn3cc(C(C)(C)N(C)C)nn3)C=CC2)=O)cccc(N)c1Br N1(C(C(C2(O)CN(C(C3(C#N)CCCO3)=O)C2)F)=O)CCC2CC1C(=O)O2 c1(C(=O)NC2(CNC(C3C(C4(C)COC4)C3)=O)CC2)cc(Cl)c(F)cc1N c1(NC(C2CCN(C(c3ccc(C)cc3Cl)=O)CC2)C)ncnc2c1cnn2C c1(CC(N2C(C)CC(C3CCCO3)C2)=O)ccccc1S(=O)(=O)N(C)CCO c1(CC(=O)N(C)CCF)cccnc1C(=O)O.c12cn(nn1)CCCS2 c1(C(=O)NCC(CCCC)NC(=O)CN2CCSCC2)nnc(O)nc1O CCCC(O)C(=O)N1CCC(C(C)(O)COC)CC1.c12ccc(s1)CNC2=O C1(OC(c2ccc(OCC)cc2)=O)CC2(C1)CC(CN)C2 C1(C(=O)NC(C2CN(C(C(=O)Nc3cccc(C)c3)C)C2)C)CC2(CCCO2)C1 c1(OCC)ccc(C=CC(=O)NCC(C(C)(C)C)NC(=O)CN(C)C)cc1 C(C(CNC(C1CCC(C)N1C(c1coc(C)c1)=O)=O)C(C)C)OC C(=O)(C(O)CCSC)N1CCC(C(=O)NC(COC)(C)C2CC2)C1 CN1CCN(C(C2CCOC(C(F)(F)F)C2)=O)C(CNC(=O)C(C)(C)CC#N)C1 C=CC(C)(O)C(=O)N1CCC(C)(NC(c2ccnnc2)=O)C1 CCS(=O)CC(=O)N1CCCC1CC(=O)NCC1CC(C)(C)CO1 c1(OC)cc(C(=O)NCC2CC2NC(c2cc(CSC)no2)=O)ccc1C C1(Nc2cc(C(N)=O)[nH]n2)CCN(C(c2ccnc(N3CCCC3)n2)=O)CC1 c1(N2CCCC(CNC(c3n(C)ccn3)=O)C2)ccn2ncc(I)c2n1 C1(CNC(C(C)N(CC)CC)=O)CC(F)CN1C(c1oc(C(C)C)nc1C)=O N1(CCC(=O)NC2CCC3CC3C2)Cc2ccccc2C1=O Cc1ccc(C(=O)NC2CCN(Cc3ncccc3C)C2)c2ccccc12 C(=O)(C(O)C(F)(F)F)N1C(C)(c2cn(C(C)CCCC=C(Cl)Cl)nn2)CCC1 N1(C(=O)NC(c2cc(F)ccn2)C(C)C)CCCC(SC(C)(C)C)C1 c1(C(=O)NC(C(C(C)C)NC(=O)C=Cc2ccoc2)C)c2c(nn1C)CCSC2 N1(C(c2cn(C)c(=O)cc2)=O)CC2(CC(NC(C3(C)COCCO3)=O)CO2)C1 Cc1noc(C)c1CNC1CN(c2cc(-c3ccccc3)ncn2)CC1F N1(C(CCC2C(C)(C)C2)=O)CC=C(C(=O)N(CCO)CCO)C1 N1(C(C(CCC)(C)CCC)=O)CCCC(C2CCN(C(c3cn[nH]c3)=O)CC2)C1 C(=O)(N=c1ncn(CC2CCCCC2)[nH]1)NC1(C)CC=CCO1 N1(C(CC(C)C2CC2)=O)CCC2CCCC12C(=O)NC1CC(CN(C)C)C1 C1(O)(CC(=O)NC(C)C(C)(C)NC(=O)Cn2nnnc2C2CC2)CCCOC1 C1(C)(C(N(C)CCNC(=O)CC2OCCC2)=O)CCSCC1.C(F)(F)F C1(C(=O)NCC(CN(C(CCSC)=O)C)(C)C)(C(=O)N(C)C)CCOCC1 C(=O)(C1CNC(=O)c2ccccc21)NC(C)CC(C)NC(=O)CSCC#N N1(C(Cc2cc(C)sc2)=O)CC2(C(=O)NCCOC3CCCC3)CCC1CC2 N1(C(CNC(CC)=O)=O)CCCN(C(=O)Cc2cc(OC)ccc2F)CC1CO N1(C(C(C)CBr)=O)CC2(C1)CN(C(=O)C=Cc1ccc(Br)s1)CC2CO c1(CNCC2(CN)CCOC2)ccc(NC(C2CNCCO2)=O)cc1 CCC(CC(=O)N1CCN(C(c2cc(C)nn2CC)=O)CC1C1CC1)C(C)C CC(C)(C)C(C)(C)C(=O)N1CC(NC(=O)Cc2ccc(F)c(Cl)c2)C(O)C1 C1(C(C)NC(C2(OC)CC2)=O)CCN(C(=O)CCC(=O)N(C)C)CC1 N1(C(CCC#CC)=O)CC(C)(C)OCC1CNC(=O)CCc1ccc(C(=O)O)[nH]1 C1(CC(=O)N(CC#C)CC#C)CCCCN1C(C1CCCC(CF)C1)=O c1(CC)cc(C(=O)N(CCNC(c2nocc2C)=O)C(C)C)cc(F)c1 C#Cc1cccc(C(=O)NC2(CC(=O)NCC3CCCCCC3)CCOCC2)c1 c1(N(C)C(C2(CNC(=O)OC(C)(C)C)CC2(C)C)=O)cccn1C1CC1 c1(CC(C)C)cc(C(N2CCCC(CN(C(=O)C3=CCSC3)C)C2)=O)cc(O)n1 c1(NC(C(CC2CN(C(CCC3CC(OC)C3)=O)C2)F)=O)cnn2c1CCCC2 C1(CNC(=O)Cn2cc(C(F)(F)F)cn2)CCC2CNCC12 Cc1oc(C)c(C(=O)N(C2CCN(C(C3CC(C4CCC4)C3)=O)CC2)C)c1C c1(NC(CC2CCN(C(c3cc(C)oc3C)=O)CC2)=O)ccc(C(C)C)cc1F c1(CCC)ccc(CC(=O)N(C(C)CCNC(c2nnc(S)n2C)=O)C)cc1 C(=O)(C(C)S(C)(=O)=O)N1CCC(CN(C(c2cnsc2C)=O)CC)CC1 Cc1nc(C(=O)NC2CC(c3ccccc3)(NC(C3(C)CCCC3)=O)C2)sc1C C1(CCNC(CC(=C=C)C)=O)CCN(C(c2nn(C)c(N)c2C)=O)C(C)C1 c1(CCC(=O)NCC(CC=C)NC(=O)Cc2cncc(C)c2)cc(F)cc(F)c1 CON(CCC(=O)NC1CCC1(C)C)C(=O)C1Cc2ccccc21 c1(CN(C(=O)C(C)Cc2cnc[nH]2)C(C)C)cccc(Cl)c1.C12CN(C1)C2=O N1(C(C=Cc2cc(C)no2)=O)CCC(CNC(C2CCCO2)=O)C1(C)C N1(CC)CC(C(N2CCN(c3nc(C)sc3C)CC2)=O)CC1=O Cc1ccccc1C1(C(=O)Nc2cccc(Cn3ccnc3)c2)CC1 CC(C)C(C(C)NC(c1cc(Cl)sc1Cl)=O)NC(c1cc[nH]n1)=O C(CC(=O)NCC(CNC(=O)COCP(C)(C)=O)CO)(C(F)(F)F)NC(C)=O C1(CCC(=O)N(CC(O)CO)C)CCN(C(=O)COC2CCC2)C1 C(=O)(CCCN(C)N=O)N1CCC(N(CC(C)C)C(c2cscn2)=O)CC1 CC(C)(C)C(CNC(C1CC(O)CN1C(C1CCC2(CCC2)C1)=O)=O)CO Cc1[nH]nc(C(=O)NCC2CCC(C)CN2C(=O)C2=CC(C)(C)C2)c1[N+](=O)[O-] c1(SCC(C(=O)N2CCOCC2)NC(C(COC)NC(C)=O)=O)ccccc1Cl C=CC(C)(C)CC(=O)N(CC(C)O)CCNC(=O)CC1COC(C)(C)CO1 C(=O)(C(C)(C)NC(=O)CC1CCCO1)N(CC=C)CCO c1(OC)cc(NCC2CCCC(NC(c3cnns3)=O)C2)nc(C(F)(F)F)n1 CC(C)C(C#N)C(=O)N1CC(O)CC1(C)C(=O)NCCOC1CC1 C1(F)(CNC(C(=O)NC(c2nc(C)[nH]n2)C)=O)CCCOC1 CC1CCCCCN1C(c1cc(Br)c(Br)n1C)C(=O)NCCCC1CC1 N1(C(C(C)OCCC(C)C)=O)C(C(N2CC(C)(F)C2)=O)CC1C c1(C(N2CCC(NC(=O)Cn3nccn3)C(F)C2)=O)cc([N+](=O)[O-])ccc1Cl C1(NC(C=C=C(C)C)=O)CCCCCCC1NC(C1(CCN=[N+]=[N-])CC1)=O c1(C(=O)NC(CCNC(C2(COC)CC2)=O)C)sc(Cc2ccccc2)nc1C N1(C(c2c(C)c[nH]c2)=O)CCOC(C(=O)NCC(C)CC2CCCC2)C1 CCC(CC)(CC)C(=O)N1CCN(C(c2ccc(Cl)c(C)c2)=O)CC(C)C1 C1(NC(C(F)=CCC)=O)CCC(CNC(c2occc2C)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(C(C)NC(C2OCC2(C)C)=O)C1 c12ccc(cc1)CC(=O)O2.N12CC(C1)C2=O.C(C(=O)NCC)=CCOC CC1CCC=C1C(=O)N1CCN(C)C(C(=O)Nc2cnccc2C2CC2)C1 Cc1cnc(C(=O)NCC2CC(NC(=O)CCC(=O)NC3CC3)C(O)C2)nc1 c1(CN2CC(NC(c3scnc3-c3ccccc3)=O)C2)cnc2n1CCOC2 Cc1ncnc(C)c1C(=O)N(C1CCN(C(=O)CCOC2CC2)C1)CCO N1(C(c2c(Cl)nc(OC)s2)=O)CCN(C(=O)C(C)N(C)C)C(CC2CC2)C1 c1(CN(C2CCCC2)Cc2cccc(OC)c2)c(Cl)cc(O)cc1Cl Cc1cc(NC(C2CN(C(c3ncccc3F)=O)CC2C)=O)c(C)cc1F c1(OC)cccc(OS(=O)(=O)CCOCCCO)c1CSC C(CCCCC(=O)N1CC(F)CC1CNC(c1cnc(C2OCCO2)s1)=O)SC c1(CCC(=O)NC2CCCN(C(c3ccccc3F)=O)C2)ccc(O)nc1 C1(C(=O)NC2CN(C(CCC(=O)NC)=O)CC2C)CCc2nnnn2C1 CC1(NC(c2cnc(-c3ccco3)s2)=O)CCN(C(=O)CNC=O)CC1 CC12CCC(C(N3C4CCC3CN(C(C35CC3CCC5(F)F)=O)C4)=O)(CC1)CO2 c1(N2CCC(C=C)C2)nc(=NCCS(C)(=O)=O)[nH]c2cc(C)ccc12 C=C(C)CC(C(=O)N1CC(C(=O)NCC2CC3CCC3C2)CC(C)C1)OC c1(N(C2CCN(C(C3N(C(CC)=O)CCC3)=O)C2)CCO)ncnc2scnc12 N1(C(CN(CCC)C)=O)CCN(C)CC1C(=O)NCC1CCC1C(C)(C)C c1(C(=O)NC(CNC(c2c(OC)cnc(Cl)c2)=O)C)ccc(Cl)c(F)c1N S(=O)(=O)(c1ccc(NC2CCCN(C)C2)c(F)c1)NCC1CC(C)C1 N1(CC(=O)Nc2c(-c3ccc(C)cc3)cccc2)C2CCCC1CC(O)C2 c1(CCC(=O)OCC)ncc(C(N2CCCC2C2(C)CC2)=O)s1 C1(CC(N2CCC(COC)(NC(=O)C=Cc3cccs3)C2)=O)OCCCC1(C)C c1(C(=O)NCC2N(C(C3N(C)C(=O)NC3)=O)CCCC2)c(O)ccc(Cl)c1F Cc1cc(C(N2CC3CC(NC(=O)C(c4cncc(F)c4)C)C2C3)=O)cc(N)c1 C(CN=C(NCC(N1CCC(CO)CC1)=O)N1CCC(O)C(C)C1)OC(C)=O C1(C(N2CCC(OCCNC(=O)Cn3cncn3)C2)=O)CCCCCS1(=O)=O n1(CCCC(=O)N(CCN(C(=O)CN2CCC2C)C(C)C)C)c(O)nnc1O C1(N(C(CCCCCn2cc(C(CC)OC)nn2)=O)C)CN2CCCCC12 C(=O)(CCCCC(N)=O)N1CCCC(CNC(C(c2ccccc2F)C)=O)CC1 C(=O)(C(F)CCC(C)C)N1CC(C(C(N2CCC(C)(COC)C2)=O)O)C1 c1(CN(CCC(CN)CO)CCC)cc(C(=O)OC)nn1C c1(C(=O)NC(CC)CNC(=O)C(C)(C)C(F)F)cc2cc(OC)cnc2[nH]1 c1(C(N(CCN(C(C2(C(=O)OCC)CC23CC3)=O)C)C)=O)ccnc2c1CCC2 CC1CN(C(=O)C=CC2CCCO2)CCCN1C(=O)CCc1ccc(Br)s1 C1(C(=O)NC2CCN(C(c3ccc(F)cc3Br)=O)C2)CC2CCCCN2C1 C1(NC(=O)CSC(F)F)CCCC(NC(c2ccncc2-n2cccn2)=O)CC1 C1(O)(NC(C(=O)NCCCN(C2CC2)CC)=O)CCCNC1 N1(C(CC=C)=O)CCC(N(C(=O)CCC2CC2(Cl)Cl)CC2CC2)CC1 c1(COC)ncc(C(=O)OC2CCCC(N(C)C)C2)c(C(F)F)n1 N1(C(=O)OCC)CCC(C(=O)NCc2cn(NC(=O)CC3CC(F)C3)nn2)CC1 c1(C(=O)NCC2C(CC(=O)NC(CCC)CO)C2)c[nH]c(C#N)c1C C1(CN(C(c2cnc3ncccn23)=O)Cc2ccco2)Cc2ccccc2O1 c1(C(C(=O)NCC2CCN(C(c3cc(C(=O)OC)no3)=O)C2)=O)ccc(Cl)cc1 N1(C(=O)C2=CCCOC2)CCC2(CC1)CC2(CO)CNC(C1(C(N)=O)CC1)=O n1(CC(N2CC(C(n3cc(-c4ccc(N)cn4)nn3)C)C2)=O)ncc2ncccc12 CCCCCCCC(F)C(=O)NC(C1CCN(C(=O)Cn2cnnc2O)CC1)C C=C=CCCC(=O)N1CC(CC(=O)N(C)CC2CC2C)C(C)C1 C(=O)(C(CCC)NC(=O)C(=O)NOC)NC(CC#C)C(=O)N1CCCC1 C1(CNC(CCC)=O)CC(C(F)(F)F)CCN1C(c1cc(Cl)nnc1O)=O C1(C2CCN(C(C3(N(C)C)CC3)=O)CC2)(NC(C2C(C)=C2)=O)CC1 C1(C(=O)NCCCP(C)(C)=O)C2CC(O)C(C2)N1C(C12CCC(C1)C2(C)C)=O CCC(C)CC(C)C(=O)N1CC(CCCCNC(C2(O)CCOCC2)=O)C1 CCCCC(C)(F)C(=O)N1CCN(C(=O)CNC(=O)CCc2nccs2)CC1 C(=O)(C(C)CNC(C1(CCF)CC1)=O)N(C)CC c1(C(=O)NC(C)CNC(=O)CCCF)ccc(C(F)(F)F)nc1O C1(NC(=O)CC2CC(F)C2)CCC(CNC(C2CC23CCCC3)=O)CC1 C1(C(=O)NC(c2onc(C)n2)C)CC(C)CCN1C(=O)CC1(N(C)C)CCC1 C1(CC(C)C)(C(=O)NC(C)CC2CN(C(C3CC=CC3)=O)C2)CCNC1=O C(=O)(CCC(CC)CC)N(CCC(=O)NCCC1CC1C(=O)OC)CC#C c1(CC)cnc(Cl)nc1NC1(CNC(=O)C(C(C)C)N(C)C)CCCCC1C C1(C(N(C(C)C)CCNC(C2CC(O)C2)=O)=O)CCCC(=O)N1 CC(C)C1=NOC(C(N2CCCC(NC(c3cccnc3C(F)F)=O)C2)=O)C1 N1(C(C)=O)CCN(C(C2CN(C(C3C4CCC(F)C34)=O)CCO2)=O)CC1 C(=O)(C(C)CCCOC)NCC1(CNC(CC=CC=C)=O)CC1 C1(C(=O)NCC#C)CC(C)CN(C(=O)CSc2ccc(F)c(F)c2)C1 N1(C(c2nc(C(C)OC)sc2)=O)CCC(NC(=O)C2=CCCS2)C12CCC2 c1(C(=O)NC2CCC(CCNC(c3scc(C(C)=O)c3)=O)C2)nc(=O)n(C)[nH]1 N1(C(C2C3CN(C(C4(C=C)CCOCC4)=O)C2C3)=O)CCC(C2CCC2)C1 C12(CNC(C3CC(=O)NC3)=O)CC(CN1C(c1ccc(Cc3nc[nH]n3)cc1)=O)C2 C1(N(C(=O)CCCn2ccnn2)C)CCN(C(=O)CN2CC(=O)NC2=O)CC1 CCCCCC=CCC(N1CCC(NC(c2ccsc2CC)=O)C1)=O c1(CC)snc(C)c1C(=O)NC1CC(CO)N(C(=O)CCNC(=O)NC)C1 C1(NC(C(C2CCCO2)CC(=O)NC2(C)CCC2)=O)CCCC2(CC1)CC2 n1(CC(N2CCCC(NC(CCC(C)CN(C)C)=O)CC2)=O)cc(F)ccc1=O CS(=O)(=O)c1csc(CNC(c2nc(C(F)(F)F)cs2)c2nnnn2CC)c1 C1(CC(C)C)CCCCN1C(C1C=CCN(C(=O)C(F)F)C1)=O CCN(CC(C)C#N)N(C)Cc1cccc(-c2ncc[nH]2)c1 c1(C(N2CCCC(CN(C(COC)=O)C)C2)=O)ccc2c(OC)nccc2c1 C(=O)(C1COc2ccccc21)NCCC(F)Cn1cc(Cc2c(C)ncs2)nn1 CCCCCCCCCCCNc1cc(NC(c2nc(CO)cs2)C)ncn1 c1(NC(c2cccc(CN3CCN(CC(F)(F)CO)CC3)n2)=O)ccc(F)cc1 n1(CC)ncnc1C(=O)NCC1C=CC(NC(=O)C(O)C2CCCC2)C1 c1(N2CCC(N(C(=O)CC3CCCCN3C)CCC)C2)ccnc(Cl)n1 c1(C(N2CC(CNC(C3(O)CCC(CC)C3)=O)(OC)C2)=O)ccc(Cl)nc1OC CC1CN(CC(=O)N(c2ccccc2)Cc2cccs2)Cc2c[nH]nc21 c1(CN(C(C2(n3cc(C(=O)OC)nn3)CC2)=O)C)ccc(C(F)(F)F)c(C)c1 c1(C(=O)NCC2(CNC(C(CCSC)O)=O)CCCC2)nsc2ccc(C)cc12 C1(NC(=O)CC2(OC)CN(C(=O)OC(C)(C)C)C2)CCOC(c2ccc(Cl)cc2)C1 CCC(C)C(O)C(C)C(=O)N1CC(F)(CNC(=O)Cc2ccn(CC)n2)C1 c1(CNC(C23CCC(OC)C2CC3)=O)ccc(O)c(F)c1F C(N=C1NC2=C(CCCC)C(=NC3CCCCC2C3)N1)c1c(CC)cccc1 C(=O)(N1CCC(C(=O)NC2CCC23CCCC3)O1)c1ccc(CC)nc1 N1(C(C2(SC)CCC2)=O)CC2CCCC(NC(c3ccn4ccccc34)=O)C2C1 N1(C(C(C(C)NC(COCC#C)=O)C)=O)CCC(C)(CO)CC1 CC(C)(C)CC(O)C(=O)NC1CCN(C(c2onc3ccccc23)=O)C12CC2 C1(C)(CNC(C(COCC)C)=O)CCN(C(C2CCC(=O)N(C)C2)=O)CC1 c1(CC(=O)NCC2CCCN(CC3CCCC(O)C3)C2)c[nH]c2cccc(F)c12 C1(C(=O)NCCN(C(c2c[nH]nc2C(C)(C)C)=O)CC)CCCC1OC Cn1c(C(=O)NC2COCC2NC(=O)Cc2cncc(F)c2)cc2sccc12 C(=O)(CCCCCCC(=O)NCC(C)NC(C1CC(=O)N(C)C1)=O)OC N1(C23C(C)OC(CO)(C2)C3)C2C=C(c3cccs3)CC1CC2 C(=O)(C#CC1CCOCC1)N1CCCCC(CCC(=O)N(CC(C)C)C)C1 c1(C(N(C(C)C)CCNC(C2CCC(C)O2)=O)=O)ccccc1-c1ncc[nH]1 c1(C(N2CCSC(C(N3CCC34CCCCC4)=O)C2)=O)sc(Br)c2c1OCCO2 C1(CNC(=O)Cc2cccnc2)CCC(NCc2cnc(C(F)(F)F)nc2)CC1 CC(C)CCCC(=O)NCC1(CCNC(c2cccc(O)c2F)=O)CC1 N1(C(CC(C)OC)=O)CC(CNC(C2(Oc3ccccc3)CC2)=O)CC1(C)C c1(CCNC(=O)NCCC2CC2(F)F)cccc(O)c1 CCC(CC)(CO)C(=O)NCC1CN(C(C2CCOC2)=O)CC1(F)F Cc1c(C(=O)NC2CN(C(=O)CCN3CCCCC3)C2)cno1 c1(C(=O)NCC(C)NC(C=C(CC)C)=O)cccc(COC)c1 Cc1ncc(NC(=O)C(CNC(=O)CC2COCC(C)O2)CC(C)C)cc1C#N N1(C(c2n(CCC)ccc2)=O)CCOC(c2ccccc2-c2nn[nH]n2)C1 C1(NC(C23N(C(C(C(C)C)F)=O)CC(C2)C3)=O)CC(C)N(C)CC1C c1(CC)cc(=NC(=O)C2(CNC(=O)COC3CCOC3)CC=CC2)[nH]n1C c1(C(=O)OCC)ccc(C(=O)NCC(C)OC)cc1.C1(C2C=N2)CCCC1 Cc1cc(Br)cnc1C(=O)NC(C1(O)CN(C(=O)C(C#N)C(C)C)C1)C C(=O)(C1CCCc2nccn21)NCC(CNC(c1onc(C)c1C)=O)S(C)(=O)=O C1(CNC(CC(=O)NC)=O)CCN(C(C2(C)CC(OC)CN2C)=O)C1(C)C CN(C)S(=O)(=O)NCC(=O)NCCC1CN(C(C2CCC=CCC2)=O)C1 c1(C(F)(F)F)ccc2ccc(NC3CSC4CCCC34)nc2c1 c1(C(=O)NC2(CNC(CC(n3c(CC)ncc3)C)=O)CCC2)[nH]c(C)cc1C Cc1nc2ccccn2c1C(=O)NC1CCCCC1N(C(=O)C(C)C(C)(C)O)C c1(-n2cc(C(C)OC)nn2)ccc2c(c1)CCN(C(=O)C(C)(C)CF)C2 c1(CC)cccnc1C(N1CC(CNC(C2COCCC2C)=O)(COC)C1)=O n1(C(C)C)ncnc1CN1CCC(CC(=O)NCCC(C)(C)O)C1 n1(CC(=O)NC(C(C)NC(c2cc(Cl)sc2Cl)=O)C)[nH]cc2c(=O)ncnc1-2 N1(C(Cc2cc(C(=O)OC)ncc2)=O)CCN(C(C23CCC(C2)C3)=O)C2CC12 Cc1ccccc1OCC(=O)NCCOCCNC(=O)CC1CC1C c1(C(C)=O)ccc(C)c(C(N2CC(C(C)NC(=O)CN3CCOC3=O)C2)=O)c1 Cc1cc(C(=O)NCC(C)N(C(=O)CCc2ccn(C)n2)C)cnn1 C1(c2ccccc2)(SC)CNC(=O)C1.C1C(C)C(=O)N2CCC2CNC1=O C1(NC(=O)Cc2cncnc2O)CS(=O)(=O)CC1NC(c1cc(CO)on1)=O c1(C(=O)NCC2CN(C(C(C(C)C)n3ccnc3)=O)C2)cc(Cl)c(Cl)cc1N c1(OC)ccc(S(=O)(=O)N2CC3CC3(NC(=O)CCCN(C)C)C2)c(Cl)c1 c1(SC)cccc(Cl)c1NC(C1CCOC(C(C)(C)C)C1)=O c1(C(N(CC(N2CCN(C(=O)C(C#N)C3CC3)CC2)=O)C)=O)c[nH]cc(Cl)c1=O N#Cc1cccc(CN(C2(CO)CCOCC2)C)c1 C12(C(=O)NCC3CCN(CCC)C3)CC(CN1C(=O)Cc1cccnc1)C2 c1(CC(=O)OC(C)(C)C)cccc(NC(N2CCCC2C2CCNC2)=O)c1 N1(C(c2c(CC)nccn2)=O)CC2CCC(C1)N2C(=O)CC(C)(O)COC c1(OCC)ccc(NC(=O)C(C)OC(=O)Cn2c(C)csc2=O)cc1 CCC(C)CC(=O)NC1CC(C)N(C(c2cncc(COC)c2)=O)C1 c1(C(N2CCN(c3c(C#CC(=O)O)cn[nH]3)CC2)=O)cc2ccccc2cn1 c1(OC)cc([N+](=O)[O-])ccc1C(N1C2CCC1CN(C(=O)CCS(C)=O)C2)=O CC1CCN(C(=O)OC(C)(C)C)CC1CNC(c1ccnc(CN(C)C)c1)=O c1(SCC(N2C3(CNC(c4c(C)nco4)=O)CC(C2)C3)=O)cc(F)cc(F)c1 N1(C(COCCCCOC)=O)CCCC1CC(=O)NCC1(O)CN(C)C1 c1(C(=O)NCCCN(C(CC(CCC)C)=O)C)ccc(S(N)(=O)=O)cc1N c1(C(N)=O)nc(C(N2CC3CC3(NC(C3CC3C(F)F)=O)C2)=O)ncc1Cl S(=O)(=O)(c1cccnc1NCC1(C)COC1)NCCC(COC)(C)C N1(C(c2cnc(C3CCC3)o2)=O)CCCCCC1CNC(C1(CCF)CCC1)=O C1(C(c2cn(CC)nn2)C)CCCCCC1.c12ncoc1C(=O)NC2(C)C CC(CCc1cccc(F)c1)C(=O)NCC(C)(C)NC(=O)Cc1nc(=N)[nH][nH]1 C1(NC(c2cc(OC)no2)=O)C=CCN(C(=O)C=C2CCN(C)CC2)C1 C(C(C)C(C)(c1nnnn1C1CCCC1)NCCc1sccc1Br)OC N1(C(C2CCCC(OC)C2)=O)CCCC(F)(CNC(=O)CCCN(C)C)CC1 O=C1CCCC(CC(=O)NC2CCCCC2CNC(=O)COc2cccnc2)N1 Cc1cn2cc(C(=O)NCC3C(C)CCCN3C(=O)CCc3cnc[nH]3)nc2s1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC(O)C1 N1(C(C(C)OCc2cccc(C)c2)=O)CCC(NC(=O)C(F)=CCCF)C(C)C1 c1(CCC)cc(C(=O)NCC2CC(O)CN2C(=O)C(C)C(F)F)c(C)o1 C1(CNC(C2N(C(C)C)CCC2)=O)CCCCN(C(=O)CCC2CCOC2)CC1 C(=O)(C#CC1CCOC1)NC(CC(C)NC(c1ncc(C(N)=O)cc1Cl)=O)C C1(C(=O)NCCNC(=O)Cc2ccc(C(F)F)cc2)CC2C=CC1CCC2 N1(C(c2c(CC)cco2)=O)CCN(C(c2ccc(C)nn2)=O)C(CC(F)(F)F)C1 c1(C(=O)NCCN(C(C)C)C(C2CCCC(N(C)C)C2)=O)ccc(N(C)C)nc1 C1(CN(C(c2cnc(O)[nH]2)=O)CC)CCN(C(C2CC(O)CN2C)=O)CC1 c1(C(=O)NC2CCC(CC(=O)NCCCC(=O)OC)C2)nc(C)c(C)s1 C1(C)(CNC(C2C(C)=CCS2)=O)CN(C(c2ccc(O)c(C)c2)=O)CCO1 N1(C(C(c2cn(CC)nc2)(F)F)=O)CC(NC(=O)CN(C)CCO)C2CC12 CS(=O)c1ccc(C(=O)NCC2CCN(C(=O)C(C3(O)CCCC3)F)CC2)cc1 C1(NC(CCOCC)=O)CN(C(c2ccc(C)c(Cl)c2F)=O)CC(F)(F)C1 CN1CCC(C)(C(N2CC(O)(C(F)C(=O)NC3CCC4(C(C)C)CC34)C2)=O)C1 CCCCCC(O)CC(=O)N1CCC(C(N2CC(O)(C3CC3)C2)=O)C1C(C)C c1(C(=O)NCC23C(CN(C(c4c(C)nc[nH]4)=O)C2)C3)[nH]c2ccccc2c1C CCC(C)(CNC(=O)CCCOC(C)(C)C)NC(c1cccn1CCN(C)C)=O Cc1ccccc1C(=O)NC1(C(=O)NCCc2cccc(O)n2)CCN(C)C1 CC(C)C(C)(C)C(=O)NCCCC1CCCN1C(C1C2CCC1CC2)=O C1(CNC(c2cccc(COC)c2)=O)CN(C)CCN1C(C1CCSC1)=O C1(NC(c2cc(C)c(C)[nH]2)=O)CC(F)CN(C(C2CC3(CCC3)CO2)=O)C1 C1C(O)CCC(=O)N1.CC(C(=O)NC1(C(N2CCCC2)=O)CC1)C1CCCC1 Cc1nnc2n1CC(C(=O)NC1CC3CCC1CC3NC(=O)C(N)=O)C2 C1(CNC(Cc2cc(C)on2)=O)CC2(CCN(C(=O)C=CC(F)F)CC2)CO1 C1(CC(=O)NCCc2nc(CC)[nH]n2)CCCN(C(C2CN(C)CCO2)=O)CC1 N1(C(C(C(C)(C)C)O)=O)CCC2OCCN(C(c3cc(CCCO)on3)=O)C2C1 c1(C(C)OCC(=O)N(CC(C)(C)ON)C)cccc(Cl)c1F c1(C(C)C)cccc(CNC(c2cnc(OC)s2)=O)n1.C(C)(C)(C)OC(=O)NC N1(C(C(C2CCOC2)NC(CC)=O)=O)CC(C)OC(C)(C)C1C N1(C(C(C2CCC2)OC)=O)CCC2CN(C(=O)CCCc3cncs3)CC2CC1 c1(C(C=CC(=O)OC(C)C(=O)NCc2ccc(Br)s2)=O)ccccc1 c1(CC)ccc(F)cc1C(=O)N(C)CC1(NC(=O)CC2CCCC(F)(F)C2)CC1 C=Cc1cncc(C(=O)NC2(C(=O)NOC(CN(C)C)C(=O)N(C)C)CC2)c1 Cc1oc(C(=O)NC2COC3C(NC(=O)C(=O)C4CC4)COC23)cc1S(N)(=O)=O c1(C(N(CCOCCNC(c2c(C)cc(F)s2)=O)C)=O)cn2cccc(Cl)c2n1 C1(c2n(Cc3nnn(C)n3)nnn2)CCCC1(CSCCCC(N)=O)NCC C=CCC(C(=O)N1CC(CNC(=O)Cc2ccc(C)o2)C1)OC C(N=c1[nH]cc2ncnc-2[nH]1)C1CCCN(C)C1=O C#Cc1ccc(CCNC(=O)C(=O)NCC2CCOC2=O)cc1 N(C(=NCCC1(C)CC1(Cl)Cl)NC1CCCCC1)C(C)C c1(C(N(C)CC2CCN(C(C(C)CO)=O)CC2)=O)nccc(N)c1Cl N1(C(CC2(OC)CC2)=O)CCOCC(CNC(C2(c3cc(C)on3)CC2)=O)C1 CN1C(=O)CCC1C(N1CCCCC1)=O.N12CCOCC1C(=O)N(C)CC2=O C1(OC)CN(C(c2ccc(C)s2)=O)CC1NC(c1nc(C)oc1C)=O C(c1nc2ccccc2o1)=CC(=O)NCC1CCCC(NC(=O)CC2(O)CC2)C1 C(C(C)(C)CC1CN(C(=O)CC2CCCCO2)C1)NC(C=C(C)Cl)=O N1(C(=O)CN2CCCCCC2)CC2(C1)CN(C(C1(c3ccco3)CC1)=O)C2 C1(NC(Cc2cc(C)on2)=O)CC2(NC(c3coc(C)n3)=O)COC1C2 c1(CC2(CC(=O)N(C)CC3CN(C(C4C(C)CCS4)=O)C3)CC2)ccccc1F N1(C(Cc2c(C)nc(C)s2)=O)CC2C3CCC(C2C1)N(C(=O)C1=CC(C)CC1)C3 Cn1cc(C2CC2C(=O)NCC2(C3CC3)CC2)cn1.C12(CC1)CCNC2=O C1(NC(c2c(C)nn(C(C)C)c2)=O)CCN(C(c2cc(Br)cn2C)=O)CC1O N1(C(C(C)S)=O)CCC(O)(CNC(c2cc(O)ccc2Cl)=O)CC1 c1(C(=O)OC)cccc(C(c2nnnn2C(C)C)NC(C)=O)c1 C(C(C)(C)C(C)(C)C)NC(C1C(CNC(CCCCOCC)=O)C1(C)C)=O c1(C(=O)NCC(CC=C)NC(=O)CC2CCCCO2)c(N)cc(OCC)cc1F C1(C(C)C)(CO)CCN(C(=O)CC(C)NC(c2cnsn2)=O)C1 CC(CCCC(=O)NC1COC(C)(C)C1)NC(c1nccnc1N)=O N1(C(CCC)=O)CCCC(C2CN(C(c3cccc(SCCC)c3)=O)C2)C1 N1(C(c2c(C)nn(C)n2)=O)CCN(C(C2COCC(C)O2)=O)C(CCO)C1 CCCCC(O)CC(=O)N1CC2CC2C1C(=O)N(C1CCC(C)(C)C1)C C(CC(C)C)(C(=O)NCC1CCCCCN1C(c1ccncc1F)=O)NC(C)=O c1(C(=O)NC2C(NC(c3cc(I)ccc3F)=O)C2)ccc(-n2cccn2)c(Cl)c1 C1(C(=O)NC23C(CN(C(CN4CC(C)C4)=O)C2)C3)CCOC2(CCCCC2)C1 c1(OC)ccc(Cl)c(C(=O)N(C2CC(NC(C3(C4CCCO4)CCC3)=O)C2)C)n1 c1(CC)c(NCC(=O)OC(C)C)cccc1C.N12CCCC1C2=O CN1CC(C(=O)NCC=CC(N2CCCCC2CCO)=O)CC1=O C=C(Cl)C(C)(C)C(=O)NC1COCC1CNC(c1cnnn1Cc1ccccc1)=O C#Cc1ccc(NC(=O)C(c2ccccc2)SCCC(C)C=C)cn1 c1(-c2cccc(C(C)C)c2)ccc(NC(c2c(F)ccc(F)c2Cl)=O)c(C#N)c1 N1(C(C(C)OC)=O)CC2CCC(NC(=O)C(C3CCCC3)OC)C2C1 C(=O)(C1=C(Cl)CCCC1)N1CC(O)(C(C(=O)NCC2(CC)CCCC2)F)C1 N1(C(CC2CC(=C)C2)=O)CCC(C2CC2)(CNC(c2ocnc2C(F)F)=O)C1 Cc1cnc(C(=O)NC23CC(C2)C3)cc1C.c12c[nH]nc1C1CCN(C1)C2=O N1(C(CCCC#C)=O)CCN(C(=O)C(N2CCOCC2=O)C)CC1CC#N C1(C(=O)NC2CN(C(c3[nH]cc(C(C(C)C)=O)c3)=O)C2)CCCCN1C1CCCC1 Cc1cc(=NC(=O)C2(C)CCCN(Cc3ccc4cc[nH]c4c3)C2)[nH]o1 Nc1cc(F)ccc1C(N1CCC(NC(c2cc(C(F)F)cs2)=O)C1)=O c1(C(N2CCN(C(C(CNC(C)=O)(C)C)=O)CC2)=O)ncnc2c1CCC2 N1(C(c2c(OC)csc2)=O)CCCC(C(=O)Nc2cccc(OC)c2)C1C N(C(=NCc1ccc(OCC(N)=O)cc1)NCCN1CCOCC1C)C1(CF)CC1 Cc1cc(CN2CCC(F)(CNC(c3cc(I)ccc3F)=O)CC2)c(F)cc1Br c1(C(N(CCCC(=O)NC(C)Cc2cccnc2)C)=O)ccc(F)nc1 CC(O)C(F)(F)C(=O)N1C(CNC(=O)C(C)(C)c2cccs2)CC2CC12 C1(CNC(C(C)CSc2ccccc2)=O)CC2CCC1N2C(=O)C(C)(F)F c1(C(=O)NCC2CCN(C(C3(CC)CCC3)=O)C2)nc(C)ccc1C C(=O)(C1=CCOCC1)NC(C(N1CCCC(CC(C)C)C1)=O)C1(C)CC1 c1(C(N2CC(CNC(=O)CC3CC(F)(F)C3)C(O)C2)=O)cc2cc(F)ccc2[nH]1 C1(C(=O)NCc2nc(CC)on2)CC2(CCC2)CN1C(C1CN(C(C)=O)C1)=O C=CCCN=C(NCC1CC(CC)C1)NCC.C1(C)C=CCCCC1 N1(C(C=CC(CC)C)=O)CCC(C(=O)NCC(C)C2CCC2)(CF)C1 O=S(=O)(c1cnccc1F)N1CCCC(c2ccccn2)C1 c1(OC)ccc(F)cc1NC(=O)CN(C1CCN(C(=O)C(O)C2CCCC2)C1)C C12(NC(CCC(=O)N(C(C)C)C)=O)CCC(C1)N(C(c1cnc(N(C)C)s1)=O)C2 C1(C(=O)NCC2C(OC)CCC2)CN(C(=O)CSC(F)F)CCC1(C)C C=CCCCC(C(=O)N(C)CC1(C#N)CC1)NC(=O)CCC1CCC1 CC1OC2(CNC(=O)CC3CC4C=CC3C4)CC1(NC(=O)Cc1cccnc1)C2 CC1=CCN(C(=O)C(c2ccccc2)NC(=O)C(C)N2CCCC2)C1 C1(CC(=O)NCCCCNC(C2(N3CCCC3)CCC2)=O)CCCOC1 Cc1cc(CCCC(=O)N(C(C)CNC(=O)C(C)Cc2ccncc2)C)c(C)s1 C(C)(C(C)(C)OCC)NC(=O)CCOCCNC(C1C(CCC)C1)=O c1(CN2CC3C(NCc4c(N(C)C)cccc4F)C3C2)ccc(C#N)c(O)c1 c1(OC)cnc(N2CCN(CC(=O)NC3CC(N4CCCC4=O)C3)CC2)nc1 N1(C(c2ncc(C)cc2F)=O)CCC2CCCC12C(=O)NCc1[nH]c(C)nc1C N1(C(c2ccc(C)cc2N)=O)CCN(C(C2CC(C)(C)C2)=O)C2CCCC12 n1(CC)nc(C)c(C(N2CCC(NC(C3CCCC4CC34)=O)C(F)C2)=O)c1Cl C1(CNC(C(C)N(CC(F)(F)F)C)=O)CN(C(=O)CN2CCC2)CC(C)(C)C1 c1(Cn2c(C(c3n(CC)ccc3)NC3CC3CC)nnn2)ccc(Cl)c(C)c1 C1(C(N2CC(C)OCC2)=O)CC(F)CN(Cc2ccc(Cl)nc2Cl)C1 N1(CC(C)C)N=C(C(=O)NCC(C)(C)NC(C2CCCC(CF)C2)=O)CCC1=O c1(C(=O)NC2C(NC(CC(CC)SC)=O)CC2)cc(OC)c(C2CC2)c(OC)c1 N1(C(C2C(C=C(C)C)C2(C)C)=O)C2CCCC1CN(C(=O)C(C)(C)F)C2 c1(C(=O)NC(C)CNC(C2CC(C)C2)=O)cc2n(n1)CC(F)C2 N1(C(CCS(=O)(=O)N(C)C)=O)CCC(NC(=O)CC2=CCCC2)C(CO)CC1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1CC(CNC(C(CC)OC)=O)C(C)(C)CC1 c1(C(=O)NCC(CN(C(c2cc(C)cc(F)c2)=O)C)O)cnc(N)c([N+](=O)[O-])c1 N1(c2c(C)cccc2)CCN(C(=O)C(O)C2(N)CC2)C(C)C1=O C(CNC(C1CCN(C)C(=O)C1)=O)(C(=O)NOCCC(O)CO)OC N1(C(c2csnc2C)C(=O)NCCCOC)CC(C)OC(C)(C)C1 C1(C(=O)NCCN(C(C2=CC(C)(CC)C2)=O)C)CC2(CCOCC2)CO1 C=C=CCCC(=O)NCc1c[nH]nc1C1CCN(C(C2CCCN2CCC)=O)C1 c1(CC(=O)NCC=CCNC(C=Cc2n(CC)ncc2)=O)csc2ccccc12 c1(C(=O)NCCCCCN(C(c2ccn(CCC)n2)=O)C)scc2c1OCCO2 c1(NC2CN(C(C(n3ncc(C)c3)C)=O)CC3C2C3)cc(C)c([N+](=O)[O-])cc1Br N1(C(c2c(CNC(Cc3cn(C)nc3)=O)occ2)=O)CC23CCC2(COC3)C1 N1(C(C2(CC)COC2)=O)CC2CCN(C(c3cccn4nnnc34)=O)CCC2C1 C1(NC(CNC(CNC(C)=O)=O)=O)CC2CC1CN(C(c1cn(C)c(C)n1)=O)C2 N1(C(C2=C(C)CC2)=O)CC(C(=O)NCC2CN(C)CCN2C)CC(C)(C)C1 C(=O)(C(F)(F)C(C)(C)O)NC(C(C)NC(=O)C(c1ccccc1)O)C c1(C(N2CC(CNC(C3=CCCC3C)=O)C2)=O)ccc2c(c1)nc(O)n2C1CC1 CCC(CC)C(C(=O)N1CCCC1CNC(=O)CCCSC)N1CCOCC1.COC C1(C(N(CCCCCNC(C(C(C)C)(C)O)=O)C)=O)C2CCC1C(F)(F)C2 Cc1cccc2c1OC(C(N1CCCCC1CN(C(=O)Cn1cccn1)C)=O)C2 c1(N(CCCN(C(C(CC)CC2CCCC2)=O)C)C)cc([N+](=O)[O-])ccc1SC N1(C(c2n[nH]c(C)c2O)=O)CCC2(CCCC2NC(c2nncs2)=O)CC1 CCC(C#N)C(=O)NC(c1cccnc1)C(=O)NCCc1ncccn1 Cc1cccc2cc(C(N3CC(C)(NC(=O)CN4CCC(C)C4)C3)=O)sc12 Cc1[nH]cc(C(=O)NC(C)(C)CNC(C2CCC(=O)O2)=O)c(=O)c1Cl N1(C(C(C)CO)=O)CCCC(C)(C)C1C(=O)NC1CCN(C)C1(C)C c1(C(N(C2CCC(NC(=O)CC=C(Cl)Cl)CC2)C)=O)ccn(C)c(=O)c1 Cc1sc(S(N)(=O)=O)cc1C(=O)NC(C)(C)C(C)NC(C1CC(C)=NO1)=O N1(C(C(C=CCCC)O)=O)CCN(C(C2CCN(C(=O)CO)CC2)=O)CC1 C1(C(N2CCC(=C)C2)=O)CCC(C)CN1C(=O)COCC(=O)NC c1(CC)ccc(C(=O)NCC(C2CCOC2)NC(=O)C(O)C(C)CC)cc1F C1(C(=O)Nc2cn(C)nc2)CCCCCCN1C(c1cc(Cl)no1)=O C1(NC(C(CCCOC)C)=O)CC2(CCCN(C(c3cccnc3C)=O)C2)C1 C1(CC)(NC(c2ccnc(C)c2N)=O)CCN(C(c2cc(C)cc(O)n2)=O)CC1 N1(C(C(CC=C)(C)C)=O)Cc2ccccc2C(NC(=O)COC2CCOCC2)C1 c1(OC)ccc(C(F)(F)F)cc1NC(N1CCCC1c1ccc(O)cc1)=O c1(SC)nc(C)c(CC(N2CC(NC(C3CCOC3)=O)C(C)C2)=O)c(O)n1 c1(CC(=O)NCC(CNC(=O)C(C)c2cccs2)OC)cc(C)cs1 c1(OCCC)cccc(C(=O)NCCC(C)N(C)C(C2(C)CCSCC2)=O)c1 C(CC(F)(F)Cn1cc(C2CCCCCC2)nn1)N(C(C(CC)O)=O)C1CC1 c1(C(N)=O)cccc(C(=O)NC2COCCC2NC(C2CC=CCC2)=O)c1 C1(C)(C(=O)N)CCCN(C(C2CC(=O)CC(=O)N2)=O)C1.C(C(C)SC(F)F)N(CC)CC CN1C(=O)NCC1C(=O)NC1CCC(CNC(c2cc(CCCO)on2)=O)CC1 C=CCC(CC(C)C)C(=O)NC1CCN(CCNC(=O)CN2CCCCC2)CC1 c1(C(=O)NCC(CNC(C(CCOC)C)=O)OC)c(C)[nH]c2ccc(OC)cc12 c1(C(=O)NCC2(CN(C(C3CC(C)OC3)=O)C)CC2)cc(O)ncc1F N1(C(C(C)OCCC=C)=O)CC(NC(=O)Cc2cncc(C)c2)C(S(C)(=O)=O)C1 CCCCC(C)C(=O)NCc1ncoc1CCNC(c1cnc(O)c(C)c1)=O N1(C(CCC(C)(C)F)=O)CCN2C(=O)C(NC(c3cc(C(F)F)no3)=O)CC2C1 C(C(CO)(CO)NC(=O)C(C(C)O)N(C)C)N(C(CC1CC(CSC)C1)=O)C N1(C(C(C)NC(N)=O)=O)CC=C(C(=O)N2CCCN(C)CC2)CC1 C1(CNC(C(C)NC(N)=O)=O)CC(O)CN1C(=O)CCCC1CCCC1 N1(C(COC)=O)CCCC(C)(C)C1CNC(C1CC1C1CC1)=O C(C(=O)NCC1(NC(=O)CCc2nc(C(F)(F)F)n[nH]2)CCC1)(C(C)C)SC N1(C(CC2NCC(C)(C)OC2)=O)CCNCC2(CCC2)C1 C(c1sccc1Br)=CC(=O)N(CC(C)NC(CCC1CC(C)C1)=O)C N1(C(C2C(C)SCCC2)=O)CC(C2CC2C(=O)NCC2(F)CC2)C1 c1(C(N(C)CC2CC(F)CN2C(=O)CC2CCCO2)=O)ccn2cncc2c1 Cc1ccc(C(N2CCC2CNC(c2c[nH]nc2-c2ccccc2)=O)=O)nc1C CC1CN(C(C2CCC(O)CC2)=O)CC(C)CN1C(=O)Cc1ncsc1Br C1(C)(C(=O)NCC(CC)NC(=O)C(F)(F)C2CCOCC2)CC2(CC2)C1 C1(C(N2CCC(O)(CNC(CSCC(N)=O)=O)CC2)=O)CCN2CCOCC12 C1(NC(CSCC=C)=O)CCN(C(=O)C=Cc2ccnn2C)CC1C(C)C c1(C(=O)NCC2(O)CCCN(C(C=CCOC)=O)C2)ccc2nc(CO)[nH]c2c1 Cc1cc(NC23C(CN(C(C4CCC4)=O)C2)C3)ncc1CNC(=O)CCN(C)C C1(NC(C2CC3CCC(C2)O3)=O)CCCCCN(C(c2cccn2C2CC2)=O)C1 Cn1nnc2cc(C(N3CC(NC(C4CC4c4cccnc4)=O)C3)=O)cnc12 CN1CCN(C(C2CC=CC(O)C2)=O)C(C(=O)NC(C(O)CO)C2CC2)C1 c1(Cn2cc(C3C(C(=O)NCC4(CF)CC4)CC3)nn2)c(F)cccc1[N+](=O)[O-] c1(C(N(C)CCC2CCN(C(=O)C3=CC(C)(C)C3)CC2)=O)ncc(C#N)cc1Cl C1(C(=O)NCC2(OC)CN(C(C3CC3(C)C)=O)C2)CC(C)(C)CO1 C#Cc1ccc(C(=O)N(CC(O)CNC(=O)CCSc2n[nH]c(C)n2)C)c(F)c1 c1(N(C)C)cc(Cl)ccc1C(=O)NC1CCC(C(=O)NCCc2cnc[nH]2)OC1 c1(COC)nc(C(=O)NC2CCC2NC(c2cc(C(=O)OC)n[nH]2)=O)cs1 c1(C(=O)NC2(CNC(C3CCCS3(=O)=O)=O)CCC2)ccncc1Cl CCCCC(C)CCC(=O)N(C(CC)CC(=O)N1CCC(C)C1)C1CC1 c1(CCC(=O)NCCCC2CCCN2C(=O)C=Cc2ccco2)cccnc1 c1(C(=O)NC2(CC(=O)NCC3(N(C)C)CCCC3)CC2)ccnnc1O c1(CC)nc(C)oc1C(N1CCC=CC1C(N1CC(OC)CC1CO)=O)=O n1(-c2ccnc(C)n2)cc(S(=O)(=O)N2C(C)CCC2C)cn1 c1(C(=O)NCCC(N2C(C(CC)C)CCC2)=O)ccc(CC(=O)OC)cc1 c1(COCC)nc(C)c(C(=O)NC2CC(NC(=O)CCOC)C2)s1 N1(C(C2(C#C)CCCC2)=O)CCC(F)(CNC(=O)Cc2cccs2)CC1 CCC(CC(=O)NCC1CC2CC2N1C(c1cnc(-c2cccs2)o1)=O)OC C1(CC(=O)NCC(C(C)O)C)CC(C)CCN1C(c1nc(Cl)cs1)=O C1(C(=O)NCC2(CC(C)C)CC2)CC(F)CN1C(C1CC1(C)C(F)F)=O C1(C(=O)OC(C)(C)C)(NC(CN(CC)CC)=O)CC(F)(F)C1.C1(C)(C(=O)NC)CC1F N1(CC(=O)NC(C2CC2C(=O)NCCc2cncs2)C)CC2CC2C1 C=CC(C)(CC)C(=O)NCC1(C(=O)NCc2ccc(OC)cc2)CC(C)(C)C1 CCCCCC(F)C(=O)N1CC(OC)CC1(C)CNC(=O)Cn1cccn1 C1(C(=O)NCC2(O)CN(Cc3ccc(C(=O)OCC)o3)C2)CCC(F)(F)C1 CS(C)(=O)=Nc1ccc(C(=O)NC2CN(C(=O)CNC=O)C3(CCC3)C2)s1 c1(OC(C)=O)cccc(C(=O)NC2CCCC(NC(=O)Cc3nc(C)no3)C2)c1 C1(OC)Cc2ccccc2N(C(c2ccc(-c3cn[nH]c3)s2)=O)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)N(CC)CC1CCCN1C(=O)C1=C(C)OCCS1 C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC2C=CC1N(C(=O)CCc1nc[nH]n1)C2 c1(C(=O)NCC2C(C)CCCN2C(=O)Cn2ccnn2)nccc2ccsc12 c1(O)cccc(Cl)n1.c1(C(=O)OCCSCCNCC)ccccc1 c1(C(=O)NCCCC(C)(C)NC(C2CCN2S(C)(=O)=O)=O)cnc2[nH]nnc2c1 CC(C)CCN=C(NCCS(=O)(=O)N(C)C)NCC1(C)CCC(=O)N1 N1(C(COC)=O)CC(C(N2CCCC2c2nncn2C)=O)C(O)C1 C(c1cnn(C)c1C)=CC(=O)NCC1N(C(C(C2CCCO2)OC)=O)CC1 C1(C(=O)NCCC(C)N2CCCC2)CC12CCN(C(=O)Cc1ccns1)C2 C(=O)(C(C)(C)CCC#N)NCc1c(CN(C(C(C)C2CCCO2)=O)C)cccc1 C1(NC(C2ON=C(C(C)(C)C)C2)=O)CCN(C(=O)C(=O)N=S(C)(C)=O)CC(O)C1 CCCCC(CC(=O)N1CCC2(CSC2)C1)NC(c1cccs1)=O CC1CCN(C(C2CCCN2C(=O)C(F)(F)F)=O)CC1CNC(=O)CC(C)(C)C C(=O)(C(C)CC(C)C(C)=O)NCC1ON=C(C(=O)NCCCCCCC#C)C1 C12(C(N(CCCCCC)CCO)=O)CCC(NC(c3cccc(=O)o3)=O)(CC1)C2 C1(CNC(CCC#CC)=O)COCCN(C(=O)C(C)N2CC(C)C2)C1 c1(C(N2CCC(CC)C2C(=O)N(C(C)C(C)SC)C)=O)cccc(C)c1N c1(C(=O)NC2CCC(n3cc(CCC(=O)NC)nn3)CC2)cc(C)cc(C)c1 c1(C(N2CCN(C(CC(C=C)C)=O)CC(C)C2)=O)cc2c(C)cccn2c1 C1(NC(C2N(C(C(CC#C)O)=O)CC2)=O)CCCCCC1C c1(OC)ccc(Cl)cc1CNC(=NCC1CC2CCC1CC2)NCC(C)(C)C C#CC1(O)CCCC(NCc2nc3ncccn3n2)C1 C1(CNC(C2(OC)CCOC2)=O)CN(C(C2CCCOC2)=O)CC(C)(C)O1 C(=O)(C(C)C(O)C(C)C)NC1C(CNC(c2ncc(C)cn2)=O)COC1 N1(C(C(C2CN(C(=O)C=Cc3cc[nH]n3)C2)OC)=O)CCC(O)(C(N)=O)C1 N1(C(C=Cc2ncc(C)[nH]2)=O)CCC(C)(C)C1C(=O)O C1(NC(c2n(CC)ccc2)=O)C2CC(NC(=O)C(n3ccnc3C)C)CC12 C1(O)(CCNC(C2N(CC)CCOC2)=O)CCCN(C(=O)C=Cc2cn[nH]c2)C1 C=CCCCCCCCC(=O)NC(CNC(=O)CCC1CCCCO1)CC N1(C(=O)NCc2ccc(-n3c(C)cc(C)n3)nc2)CCC(C2CCCC2)C1 c1(C(=O)NC(c2ccccc2)C(C)NC(C(C)=CC)=O)c[nH]c(C(=O)NC)c1 C1(CC)CC(C(C(=O)NCCC(=O)OC(C)C)N(CC(=O)OC)CC(F)F)C1 C1(NC(CC2CC(C)C2)=O)CCC(F)(CNC(=O)Cc2nc[nH]n2)C1 Cc1nc(Cn2cccn2)ccc1-c1nc(C2CC2)nn1Cc1ccc(Br)cc1 C1(CNC(C2(N(C)C)CC2)=O)CCCCN1C(=O)CCc1cccnc1 C1(NC(CS(=O)(=O)NCC)=O)CN(C(c2ccc(CC(C)C)s2)=O)CCC1C C1(O)(CNC(=O)CCCc2cccc(Cl)c2)CCCN(C(c2cocn2)=O)CC1 C#CCC(CC(=O)NC(C#C)C(C)(C)C)NC(C1CCC(=O)N(C)C1)=O C(CC1=CCN(C(C2(C)CCCO2)=O)CC1)NC(C1N(C(C)C)C(=O)CC1)=O N1(C(C2CCC(=O)C2)=O)CCCN(C(C23CCC(CC2)C3)=O)C(CO)C1 N1(C(COCC(=C)C)=O)CC(C(N2CC(=O)NC(=O)C2)=O)OC(C)C1 Cc1ccc(C(=O)NCc2ccoc2C(=O)N(C2CCOC2)CCF)cc1C CCCC(C)(C)C(=O)N1CCC1CNC(c1cccn(C(C)(C)COC)c1=O)=O c1(C(N(CC(F)F)CCOC)=O)oc(CNC(c2cnsc2)=O)nc1C C1(C(=O)NC(CC(=O)NCCCC(C)CO)C2CC2)NC(=O)OC1(C)C c1(CC(N2CC(C)(NC(CC(C)n3cccn3)=O)C2)=O)cn2c(n1)CCCC2 CC#CCC(C(=O)N(C)Cc1cnc(C)o1)NC(=O)C(C)CC CC1(C)CCC(CC(=O)N(CCC(=O)NCC2(C)CCCO2)CCCO)O1 c1(C(CC)O)nc(CCCN(C)C(C)C)n(-c2ccc(C3CC3)cc2)n1 C12(NC(c3ncc(F)cc3F)=O)CCN(C(=O)C=CSc3ccccc3)CC1C2 C12(C(N(CC(CCC)O)C)=O)CCCC1CCN2C(c1ccc(CC)cc1)=O C(=O)(CCCCC(F)(F)F)NCC1CCN(C(C(CC(=C)C)C)=O)C1(C)C c1(C(N(CCCNCC(=O)NC)CC)=O)n[nH]c(C)c1C(N1CCCCCC1)=O c1(OC)cccc(CN2CCCC(C(=O)NC3COCC3O)CC2)c1C C(CCCC(=O)NCC1CC(OC)CN1C(C1CC1C)=O)OCCC=C c1(C(=O)NC2C(O)CCN(C(c3nc(CC)on3)=O)C2)cc(Cl)cc(Cl)c1N c1(N(S(CC)(=O)=O)CCC)ncc(F)cc1C.c1(-n2c(=O)c2=O)cncnc1O C1(CNC(C(C=C)CC)=O)CN(C(=O)Cc2c[nH]c3cnccc23)CCC1(C)C Cc1cc(CCCC(=O)NCC2(NC(c3cnc(Cl)[nH]3)=O)CCC2)c(C)s1 C1(C)(CC)CC(NC(=O)CSCCN(C)C)CN1C(c1ccc(C2CC2)o1)=O C1(CNC(CS(CC)(=O)=O)=O)CN(C(=O)CC2COC(C)(C)O2)C2COCC2O1 CCC(C)(CC(=O)N1CC(O)(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)C1)C(=O)OC N1(C(c2nc(CCCCC)sc2)=O)CC(CNC(=O)C=CSC)C(C)C1 C1(C(=O)NC(CCC)C(F)(F)F)CCC(C)(C)N(C(=O)CC2CC3(CC3)C2)C1 c1(NC(C(c2ccccc2)OC(CC=CCC)=O)=O)ccccc1[N+](=O)[O-] C(C)(C)(CCCNC(C1CC2CCCC12)=O)NC(CN(C)C(=O)C1CC1)=O c1(C(=O)NCCN(C(C2CCC(O)C2)=O)Cc2ccccc2)cnc(O)c(F)c1 c1(-c2cn(CC(C)C)nc2)ccc2nc(CC(=O)NCC(O)CO)cn2c1 CC1CCN(C(=O)C(C)c2cccs2)CCN1C(=O)Cn1ccccc1=O C(=O)(CC(C(F)(F)F)NC(c1cn(C)nn1)=O)NC(COC)(C)C c1(C(N(C2(C)CCN2c2ccnc(N3CCCC3)n2)C)=O)ccc(Cl)c(F)c1 c1(CC)cc(C(N2CCC(O)(CCNC(=O)CN3CC=CC3)CC2)=O)cc(F)c1 c1(CC)cc(Nc2snc(C)c2C#N)cc(CSC)c1 CCCCC(F)C(=O)N(C1CN(C(=O)Cc2scnc2C)CC1(C)C)C C12(C(N3CCC(C)(CNC(=O)CCc4ccccn4)C3)=O)CCC(C1)C(C)(C)O2 Cc1ncc2c(n1)CCC(NC(C1OCCOC1(C)C)C)C2 N1(C(=O)NC(C2CCCS2)=O)CC2(C)CC1C2Cc1cccc(C)c1 c1(NC(=O)NC2C(CC(C)C)CC2)cnn(C(C)(C)C)c1 c1(OC)ccc(CC2(C(F)F)CC2)cc1NC(=O)NOCc1ccccc1 C1(OC)CC(CN)N(C(C2(c3ncco3)CCCC2)=O)C1 Cc1cc(=O)ccn1CC(=O)NC(C1CN(C(C23CCC(CC2)CO3)=O)C1)C N1(C(CC2(OC)CC2)=O)CCC(C2(O)CCN(C(=O)CC3C=CCC3)C2)CC1 C(=O)(C(F)C(C)(F)F)NCC1C(C(=O)NC(CC(=O)OC)C2CC2)CCO1 C1(C(=O)NCC(C)N(C)C(c2cc(C3CC3)[nH]n2)=O)COCCN1C c1(C(=O)NCCC2(O)CN(C(Cc3c(C)scc3)=O)C2)ccc2nn[nH]c2c1 Cc1cccc2c1CCOC2C(=O)N1CCN(C)C(CF)C1.C C1(NC(c2nccnc2Cl)=O)CC2CN(C(c3cc(Cl)sc3Cl)=O)CC12 C1(OC)CCCC(CC(=O)NC(C)(C)CCNC(c2ocnc2C(F)F)=O)C1 CN1CCC(C(=O)NC2CCCC2NC(c2ccnc(CC(F)(F)F)n2)=O)C1=O CC(C)(COCC(F)F)C(=O)NCC1CC1NC(C1CCSCC1)=O c1(CC)cc(C(=O)NCC2CCN(C(C3(C)CC=CCO3)=O)C2)c(C)nn1 O=C(Cn1ccnc1)NN1CCCC1C(=O)NC1CCCC(O)CC1 c1(C(=O)NCC(C)(C)CO)ccc(CN2CC3CCC3C2)cc1 CCC1=C(C(=O)N(CC(C)NC(c2[nH]ccc(=O)c2C)=O)CC)CCCO1 CCCC(C(O)C(=O)NCC1CC1c1ccco1)NC(C1CCC2(CC2)C1)=O c1(C(=O)NCC2N(C(C(CC#C)C3CC3)=O)CC=C2)cccc2ncnc(O)c12 c1(C(=O)NC2CCN(C(C3C(=C)C3)=O)CC2O)ccc(S(=O)(=O)NC)nc1 C1(NC(CCCOC)=O)COCCC1NC(c1ccncc1Br)=O C1(CNC(C2C(C(N)=O)C2)=O)CC2CN(C(c3n[nH]c(C4CC4)n3)=O)CC12 c1(C(=O)NCC(C)CN(C(=O)CCCC2CCCO2)C)cncn(C)c1=O C(CC(=O)NC(C)(CO)C1CC1)(C(F)F)NC(c1ccc(CC)[nH]1)=O CC1(C)CN(CCO)CCC1NC.c1(NC(=O)COCC(F)F)cncc(Cl)n1 C1(CNC(Cc2c(C)n[nH]c2)=O)CCCN(C(=O)CC2COC(=O)N2)CC1 S(=O)(=O)(c1cccs1)N(C1COCCN1)CC(=O)NCCCn1c(C)cc(C)n1 c1(C=O)cnc(OCCO)cn1.C12(COCC(N3CCC3CSC)=O)CCC(C1)OC2 C(C(=O)N1CC(C)(C)C1Cn1cc(CC(O)CN(C)C)nn1)(C(C)(C)C)OC N1(CC)C2CCC1CN(C(=O)CCCCNC(c1cncs1)=O)C2 N1(C(C(CNC(C2(COC)CCCC2)=O)C(C)C)=O)CCC2(CCCN2C)C1 CCC(C)CC(C)N(C)C(C1(NC(=O)CC2CCCC23CC3)CCCCC1)=O CCC(C)(CCC(C)C)C(=O)NCCC1CCCN1C(=O)CSCCC(C)C c1(CNC(c2cc3occc3s2)=O)nc2c(s1)CN(C(C1CCSC1)=O)CC2 C(=O)(C(CCCO)c1ccccc1)N1CCCC(CNC(=O)CC2(CO)CC2)C1 c1(C(N(C2CCN(C(c3ccc(CCC)s3)=O)CC2)CC#C)=O)cccc(O)n1 c1(CC(=O)NCc2c(NC(CCCOCCOC)=O)c[nH]n2)sc(C2CC2)nc1C CC1(C)Cc2nc(C(=O)NCCN(C(=O)CS(N)(=O)=O)C3CC3)ccc2CCO1 N1(C(CCSC)=O)CCC(N(C)C(C2COCCN2C(C)=O)=O)C2(CC2)C1 c1(CN2CCC(F)(CNC(C3N(C)C(=O)CC3)=O)CC2)nccc2nc[nH]c12 c1(C(N2CC(O)(CCNC(C(CC)(F)F)=O)C2)=O)cnc(SC2CC2)nc1C c1(OC)ccc(F)c(C(=O)NC2CC(NC(=O)CC(C)C)C2)c1F Cc1ccc(CC(N2CC(NC(C3(C#N)CCCO3)=O)C(C)C2)=O)c(C)c1 Cc1noc(S)n1.C(C)(C(C)(C)NC(C1(CNC(N)=O)CC1)=O)NC(CCCN)=O C(=O)(C(CC(N)=O)NC(c1ccc(C)n1C)=O)NCC(CC=C)(C)O C1(C(=O)NCC2CC(NC(=O)CCc3nccs3)C2)CCC2C(C1)C2(F)F C1(NC(c2c(C)[nH]nc2C(C)C)=O)CCCN(C(=O)C2=CCCCC2)CCC1 CC(C(=O)NCC1(CNC(C2(C#N)CC3CC3C2)=O)CCC1)C(F)(F)C(F)F N1(C(CCOCC(C)C)=O)CCC(C)(CCNC(=O)CCCCC2CC2)C1 Cc1ccc(I)c(C(=O)NCCCC2CC=CC2)c1 C(C)(C)(CC=CC(=O)NC1CC(NC(N)=O)C1)NC(CC1C(CC)C1)=O C(CC1=CCN(C(=O)Cn2cc(C)ccc2=O)CC1)NC(C1(OC)CCOC1)=O c1(C(=O)OCC(CNC(=O)OC(C)(C)C)=O)oc(Br)nc1C(F)(F)F C1(NC(CC=CC(C)(C)C)=O)CCCC1NC(=O)CCc1cscn1 O=C(C1=C(Cl)CCCC1)NCC1CC1NC(C1(c2ccccc2)CCOC1)=O C(=O)(C1=NNC(=O)C1)NCCSCC(=O)NCC(CCC)OC N1(C(C2C(C(=O)OCC)C2)=O)CCCC(NC(C23CCC(CC2)OC3)=O)C1C C1(O)(CC(=O)NCC(CC)(C)CC(N2CC(CSC)C2)=O)CCCCCC1 c1(C(N2CC3C(C(=O)NCc4n(C)ncc4)C3C2)=O)c(Br)ccc2c1OCO2 c1(CNCc2cncc(C(F)(F)F)n2)sc2c(c1I)CNC2 N(C1CC(C)n2ccnc21)C(=O)NCc1cccc(-n2ccc(C)n2)c1C C1(C(N(CCCCCC)C)=O)C2CC(O)C(C2)N1C(c1ccc(C)nn1)=O N1(C(CC(n2c(CC)ncc2)C)=O)CCN(C(c2cc(C)oc2C)=O)CC1 O=C(C1CCc2c[nH]nc21)Nc1ccc(-n2cccn2)c(F)c1 C(=O)(CCCC(=O)N(C1CCCCC1NC(C1C=CCC1)=O)CC)N(CC)CC CC(C)C(CNC(=O)CC1CCCOC1)C(=O)NCCC1CC(F)C1 C1(CNC(=O)CC2CCOC2)OCCC1C(=O)N(C1CC1)CC1CC1 Cc1cc(CN(C2CCN(C(=O)COC3CCOCC3)CC2)C)cc(F)c1 N1(C(CC(C=C)CC)=O)CC2CCCC(NC(=O)C(c3ccc(CC)s3)=O)C2C1 N1(C(C2(c3cccc(OC)c3)CCC2)=O)CC2(CC(NC(=O)CNC=O)C2)C1 c1(CC)ncc(C(=O)NCC2CCCC2NC(c2cccn2C)=O)s1 CC(C)(C)CC(O)C(=O)NCC(c1ccc(F)cc1)NC(=O)C(F)C(C)(F)F c1(C(=O)NCC(=C)CCNC(C2CC(=O)N(C)C2)=O)cnc2c(c1)CCCC2 N1(C(CN(CCC)C)=O)CCCCC1CNC(=O)C(=O)C=Cc1cccs1 C=CC(C)(CCOC)C(=O)NCc1nc(CNC(C2CN(CC)C(=O)N2)=O)cs1 C1(CO)CC(O)CN1N(CCc1ccc(F)cc1F)C1CC1 N1(C(C(C)OCC)=O)CCOC2(CCC(NC(=O)C(C)C(O)C(C)CC)CC2)C1 N1(C(c2cccnc2SC(F)F)=O)CC2(C1)CN(C(C1CCCC(F)(F)C1)=O)C2 CCC(C)(O)C(=O)NCC1(O)CCN(C(c2ccccc2-c2nncn2C)=O)C1 C(=O)(C(CC(C)(C)C)NC(=O)CCN1CCCC1=O)N(CC=C)CC=C C(CC)(C(=O)NCC(=C1CN(C(=O)C2=CCC2)C1)F)OCC c1(C(N(CCCN(C(=O)Cc2ccc(F)cn2)C)C)=O)c(S(N)(=O)=O)cnn1C C1(O)(C(N2CC(C)C(NC(C3CCCC(C)(C)O3)=O)CC2)=O)CN2CCC1CC2 c1(C(N2CCC(C)(NC(=O)C(F)=C3CCCC3)C2)=O)ccnc2c(F)cccc12 c1(NC(=O)NCCC23CCCC2C3)cccc(COc2ccccc2Cl)n1 C(CC(=O)NCCCn1cc(C)cn1)(C(C)(C)C)NC(COC(CC)C)=O CC1(C)C(NC(=O)NCc2noc(C(F)F)n2)CC1O C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(C(=O)NCC(O)CN(C)C)(OC)CC1 N1(C(C(C(C)O)NC(=O)OC(C)(C)C)=O)CC(C)(C)OCC1C(=O)O C1(C(=O)NCC2CC2NC(C2(n3ccnn3)CC2)=O)CCc2ccccc2CC1 N(C(=NCC1CCC1)NCC1CCC1)CC1C(=O)OCC1.C1(C)CCCO1 c1(NC2CCN(C(CC)C)CC2)nccc(=NCC(C)(C)N2CCCC2)[nH]1 N1(C(C(CC=CC)NC(=O)CCc2nc(O)n[nH]2)=O)CCC12CN(C)C2 N#Cc1ccnc(NC(c2n[nH]cc2NCc2cc(-c3ccccc3)no2)=O)n1 c1(C(=O)NCC(C)N(C(C2C(C(=O)OC)CC2)=O)C)ccc(C)cc1C Cc1cc(C)c(C(=O)NCC2CC3CC3N2C(=O)C(C)Cc2ccco2)c(S)n1 C(=O)(CC(C)C(C)(C)C)NC1CN(C(c2cc(C(N)=O)cc(C)c2)=O)C(CO)C1 c1(CC)cncc(C(=O)NC(CCOC)C(=O)N2CCC(CC(F)F)C2)c1.CCS C(=O)(C(C)(C)C(=O)NC(CNC(=O)CC(=O)N(C)C)CC(F)(F)F)OCC C1(CNC(C2CCCO2)=O)CCC12CCN(C(=O)CCn1ccnn1)CC2 N1(C(C(C)CO)=O)CCCC(C)(CNC(c2cccc(F)c2)=O)C1 N1(CC)CCN(C(=O)NC2CCC(c3ccc(C)cc3)C2)C(C)(C)C1 c1(C(=O)NC2CC(C)(NC(C(C(C=C)C)C)=O)C2)[nH]cc2c1CCS2(=O)=O c1(C(=O)NCC2CN(C(C3(C)CCCCO3)=O)CC2O)cccc2nccn12 C1(CC)CN(C(c2csc(Cl)n2)=O)CCN1C(C1C2CC(=O)CC12)=O C=CC1(C(=O)NCCC(O)CCC)CCN(C(=O)C=Cc2ccnn2C)CC1 Cc1ccc(C)c(C(N2CCC2(C)CC(=O)NCCC2CCCN2C)=O)n1 c1(NC(C23C(CN(C(CC(CC)O)=O)C2)C3)=O)cnc(Cl)c(Cl)c1 c1(C(=O)NC2CCN(C(C3(C=C)CCC3)=O)CC2O)cn2cc(C)sc2n1 n1(CC(=O)N(C)CC2CN(C(c3ccc(F)nc3)=O)C2)cc([N+](=O)[O-])cn1 c1(C(=O)NC(CN(c2nccc(CC(=O)OC)n2)C)C)cc(C)cc(F)c1 CC(C)(C)C(CNC(C1CC(CNC(c2ccnnc2)=O)C1)=O)CO CC(CC(=O)N1CC(C)(NC(=O)C(c2ccc(F)cc2)=O)C1)C(F)F C1(C(C)C)C(C(=O)N(CCCC(C)(F)F)C)CCN1C(=O)CCC1CCCC1 c1(C(N2CC(OC)(CNC(c3nc(Cl)cs3)=O)C2)=O)ccc2c(c1)CC(C)(C)O2 C1(CNC(c2ccc3ocnc3c2)=O)CC2COCC2N1C(c1ccncc1)=O N1(C(C2OCCN(C)C2)=O)CC(N(C)C(c2cn3c(n2)CCC3)=O)C(C)(C)C1 CN=c1ccc(C(=O)NOCC(N2CC(O)(C3CC3)C2)=O)c[nH]1 C#CC(C)(C)C(=O)NCCCC(C)NC(=O)C#CCc1ccccc1 N1(C(C2C(CC)N(C)CC2)=O)CCCOC(CCNC(c2[nH]c(C)cc2C)=O)C1 CCS(=O)(=O)CC=CCNC(=O)C(n1cc(Br)cn1)F N1(CC(=O)N(C(C2C(C)C2(F)F)=O)CC)CCC(NC(C)C)CC1 C(N=c1nnn(C)[nH]1)C1CCCC(CNC(COc2c(C(C)=O)cccc2)=O)C1 N1(c2cc(NCC3(CF)CC(F)(F)C3)nc(COC)n2)Cc2ccncc2C1 C(CCOCCO)(C(=O)NC1(C)CC(C)(C)C1)NC(C(F)=C(C)C)=O C1(NC(CC2OCC(C)(C)OC2)=O)CC2CC1CN(C(c1ccc(=O)oc1)=O)C2 N1(C(C(F)=C(C)C)=O)CCCC12CCN(C(C1CC(=C3CC3)C1)=O)CC2 N1(CCC2C(C)(C)CCC2)CCN2c3ccccc3CCC2C1 Cc1cc(C)c(C(=O)NC23CC(NC(C4CC4c4ccccc4)=O)(C2)C3)o1 CS(=O)(=O)CCC(=O)NCc1ncccc1C(=O)NOCC1CCCC1 C1(C(=O)NC(C(C)C)CNC(=O)Cn2ccc(C(F)(F)F)n2)CC(C)(C)CN1C c1(OCCC#C)ccc(C(=O)NCC(O)CN(C(=O)CC2C=CCCC2)C)cc1 N1(C(CNS(N)(=O)=O)=O)CCC2C(CCCN2C(C2CN(C(=O)N(C)C)C2)=O)C1 N1(C(CC=CCC)=O)CC2CC1C2C(=O)NCCCCCCC1CC1 c1(C(N2C(CNC(=O)CC(F)(F)F)CC(C)(C)C2)=O)cc2n(c1)CCOC2 Cc1ccn(C)c1C(=O)N(CCC(C)(C)NC(C1CC1(C)C(F)F)=O)C c1(C(=O)NC2C(C)CN(C(C3(N=[N+]=[N-])CC3)=O)C2)cccc(C(F)(F)F)c1F N1(C(C(CC)N(C)C)=O)CC2CCC(CNC(c3cn(C)c(C)n3)=O)(C2)C1 C1(OC)CN(C(=O)C(O)CNC(c2ccc(CC#N)cc2)=O)CC1O C1(C(N(CCC(=O)NCc2cc(C(C)C)on2)CC2CC2)=O)CCN(C)C(=O)C1 c1(OC)ccc(NC(=O)CCC2(C)N=N2)cc1S(=O)(=O)Nc1c(F)cccc1Br N1(C(C(C)NC(CC)=O)=O)CCC(O)(CCNC(c2oc(CO)nc2C)=O)CC1 C1(CNC(C(C)(Cl)Cl)=O)CC2(CCN(C(c3cccc(F)c3O)=O)C2)CO1 C(=O)(C(C(C)NC(=O)C1=C(C)OCC1)C(C)C)N1CCOCC(CC)C1 C1(NC(C(COC)Cc2cccc(OC)c2)=O)CNC(=O)C12CC2 C(C(C)CS(C)(=O)=O)N(C(=O)CCn1cccn1)CCCOC N1(C(c2cc(C)ns2)=O)CC=C(CCNC(=O)C(c2ccccc2)N(C)C)CC1 C1(C(=O)NC(C2CCN(C(C3(O)CCSCC3)=O)C2)C)CC2CCC(C1)S2 N1(C(c2nc(C)sc2)=O)CC2CC2(C(=O)Nc2cnn(-c3ccccc3Cl)c2)C1 c1(CC)cn2c(n1)CC(C(=O)NCC1CN(C(=O)C(C)Cn3cccn3)C1)CC2 C(CC(=O)NCCCCNC(c1nnn2c1CCC2)=O)(C(F)(F)F)OC CC(CC(=O)N1CCOC(C(C)NC(c2cnn(CCF)c2)=O)C1)C(F)F CC(C)CC(C)CC(=O)NCC1CC12CCN(C(=O)C=CC(C)(C)C)CC2 C(=O)(C(C(C)C)NC(=O)C(CCc1ccc(F)cc1)N1CCCC(O)C1)OC C(=O)(C(COC)NC(=O)CCc1ccoc1)N(CC#C)CCOC Cc1ccncc1-n1cc(CCCOCCNC(c2cn(C)nc2C)=O)nn1 N1(C(C2(OC)CCCC2)=O)CC2CCN(C(=O)CCc3cc(C)cc(C)c3)C2C1 C1(CNC(c2cnn(C3CCC3)c2)=O)CC(F)(CNC(C23CC(F)(C2)C3)=O)C1 C1(C(N(CC(CN(C)C(c2nccnc2O)=O)O)C)=O)CCCCC(C)(C)C1 C1(F)(CNC(C=CC(=O)OCCCC)=O)CN(C(c2nnn(C(C)(C)C)n2)=O)C1 N1(C(CC(C)CF)=O)CCN(C(=O)CCc2ccccn2)CC1c1ccccn1 CCC(C)C(O)C(C)C(=O)NC1C2CC3C(C2)C13C(=O)NCC1CC2(CCC2)C1 c1(C(=O)NC(C2CN(C(CCNC(=O)NC)=O)C2)C)cncc2c1CCCC2 N#CC1(C(N2CCC(CNC(C3CC3F)=O)CC2)=O)CCSCC1 C1(O)(C(C)C)CCCN(C(=O)C(C)N(C)C)C1.C1(=O)CCCC(=O)N1 c1(CNC(C(C)SCCCC)=O)c[nH]nc1C(=O)NCC(C)C(C)SC C1(CC=C)(C(=O)NCC(C)CNC(c2nc(=O)n(C)[nH]2)=O)CCOCC1 N1(C(=O)CCC2CCCC2)CCCCC(NC(C23CCC(CC2)CO3)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CCC12CN(C(=O)CSCC(C)C)C2 c1(C(=O)NC)cc(F)ccc1OC.C(=O)(C(F)=CCCC(C)=CC=C)N N1(C(C(CCNC(C(C)C2CC2)=O)(C)C)=O)C2CCC1CC1(C2)N=N1 Cc1nccn1C(C)C(=O)N1CC(CC(C)NC(=O)CC2CCOCC2)C1 c1(CNC2C=CC(CN)OC2)cc(Cl)cnc1O.C12CCN(CC1)Cc1cn2nn1 c1(C(N(c2cc(Br)ccc2I)C)=O)ccnc2c1CNCC2 c1(OCC)ccc(C(N2CC3(C2)CN(C(c2ccc(C(F)F)o2)=O)C3)=O)cc1C C1(CCNC(CN(CCC#C)C)=O)CCN(C(=O)C(CO)N(C)C)C1 N1(C(C(c2ccc(C)s2)C)=O)CC(C2CCCN(C(=O)CN3CC(C)(C)C3)C2)C1 c1(SC)ccccc1NC(=O)C(N1CCCC(c2cn(C)nn2)C1)C C#CCC(CC#C)C(=O)NCC(CNC(C1CC(OCC)C1)=O)CO c1(C(N2CCCC(CN(C(c3cc(C)no3)=O)C)C2)=O)cc2cccc(O)c2[nH]1 O=C(C1=CCCS1)NCCNC(C1CN(C(C2C3CCCC23)=O)C1)=O C1(NC(COCCC)=O)CS(=O)(=O)CC1NC(c1cncnc1C)=O CC(N=c1[nH]c2c(c(=NCc3nc4ccccc4[nH]3)[nH]1)CCC2)c1nc(=N)[nH][nH]1 c12cnccc1N(C(C)C(=O)NC(C)C(=O)NCC)C(=O)C2.CCCOC C(C(O)C(F)(F)F)N(C)C(C1(N(C(=O)C(F)(F)C2CC2)C2CC2)CCC1)=O C(C(CC)CCO)NC(CCN(CC#C)C(c1cnn(C)c1C)=O)=O c1(N(CC(C)NC(C2C(=C)CC2)=O)C)nc(C)nc(=N)[nH]1 C1(C(=O)NC2CCC(NC(CC(CCSC)O)=O)CC2)CCc2ncnn2C1 CC1CC(C)(C(=O)NCC(C)(C)CNC(=O)C=C2CCCC2)CCO1 N1(C(CCOCCC)=O)CCC2CN(C(=O)C(O)C(C)C)CC2C1 C(CN=c1nc(N2CCOC(C3CC3)C2)c2c(F)cccc2[nH]1)c1c(C)ocn1 N1(C(CC(=O)OC)=O)CCC(NC(c2csc(O)n2)=O)C12CCCC2 N(C1CCC(Nc2nccn3nccc23)c2ccccc21)C(=O)OC(C)(C)C CC(C)(O)CC(=O)N1CCN(C2CCC(NC(c3ccon3)=O)C2)CC1 c1(C(N2CCC(NC(C(F)=C(C)C)=O)C2C(C)C)=O)cc(F)c(F)c(Cl)c1F c1(C(=O)NCC(CO)NC(c2c(CC)noc2)=O)cc(C)c(=O)n(C)c1 Cc1nc(SCC(=O)OCC(=O)Nc2c(O)ccc(F)c2Br)c(C#N)c(C)c1C CC1(C)COCCC1C=CC(=O)NC1CC2CC(NC(c3cccs3)=O)CC12 C1(NC(C)=O)CS(=O)(=O)C12CCN(C(C1CC(F)(F)C1)=O)CC2 N#Cc1ccc(CC(=O)NC2CC2C(=O)Nc2cccc(CNOC)c2)cc1 N1(C(C2(C)CCC(=O)N2)=O)CCCN(C(C2CC(O)(C(F)(F)F)C2)=O)CCC1 Cc1ccc(OC(C)C(N2CCC(C(=O)NC3(C)CC3)C2)=O)c(Br)c1 CCN=c1[nH]c(C)c(C(=O)NC(C)(C)CCCNC(c2cn3c(n2)CCC3)=O)s1 Cc1ncc(C=CC(=O)NC2CCC2NC(c2ccccc2C(C)C)=O)s1 O=S(=O)(c1ccc2[nH]c(=NCCCC3CCC3)sc2c1)NCC1CC1(Cl)Cl CS(C)(=O)=NC(=O)C(=O)N1CC2CC(NC(C3CC34CCC4)=O)CC1C2 c1(CC(C)N(C)C(c2cn(CC3CCCOC3)nn2)=O)ccccn1 c1(CC)ccccc1CC(=O)NCC1(OC)CN(C(=O)CCCOC(C)=O)C1 C1(F)(C(=O)NCC2CC(CF)C2)CCC(CNC(C2(C(C)C)CC2)=O)C1 CC(C)(C)CC(O)C(=O)NC1CCC(NC(C2CC3(CCCC3)C2)=O)C1 c1(N2CC(C)C2)ccc(C#N)nn1.C(=O)(CCC1CCCO1)NC(C1CNC1)C c1(C(C)C)ccc(NC2CCC3(CN(S(=O)(=O)CC4CCC4)C3)C2)c(C#N)c1 c1(OC)cccc2cc(-c3ccc(C(N)=O)cc3)[nH]c12.N12CCC1C2 N1(C(C(F)=C(C)C)=O)CC(NC(c2oc(Br)nc2C(F)(F)F)=O)C(C)C1 O=C(CS(=O)(=O)C1CC1)N(C1CC1)CC1CN(C(=O)CC2CCOCC2)CCO1 C1(NC(=O)CCc2ccco2)CN(C(=O)Cc2ccns2)CC1C1CC1 C1(OC)(CNC(C2(CO)CC(C)(C)C2)=O)CCN(C(=O)C=Cc2ccc[nH]2)CC1 c1(CC)ncc(C(=O)NC2(CCNC(=O)C=C3CCC3)CCCC2)o1 C1(C(=O)Oc2ccc(O)cc2)(NC(c2nnnn2C)C)CCCC1C C1(C(=O)NCC(C(=O)N(CC#C)C2CC2)N(C)C)CC(O)(C#C)C1 N1(C(c2c(C)[nH]nc2Cl)=O)CCC(C2(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)CC1 N1(C(C=CCC(C)(C)NC(=O)CC(C)(C)C)=O)CC2CCOCC2C1 C(=O)(CC(C(F)(F)F)NC(=O)C1=CCCCCC1)NC(C(C)O)(C)C C#Cc1cccc(C(=O)NCC23CCC2CCN3C(c2cc(C)on2)=O)c1F N1(C(c2cc(C)nnc2)=O)CC(C(=O)NC(C(N)=O)C2CCCC2)CC(C)(C)C1 CCC(C)(CCNC(=O)C(c1cncn1C)O)NC(c1[nH]cc(C)c1C)=O CC(C)CC(F)(F)C(=O)N1CCCC(CCNC(=O)CSCC(F)F)C1 Cc1cnc(NCC2CCC=CO2)c(S(=O)(=O)NCC2(C)CCCC(=O)N2)c1 Cc1ccnc(C(N2CCC(CCCNC(=O)COc3ccsn3)CC2)=O)c1O C(c1ccc(F)cc1)=CCC(=O)NC1CC1CNC(c1ccnc(CO)c1)=O C1(CNC(C(CC=C)OC)=O)CN(C(c2cnncc2O)=O)CCC1C N1(C(c2scc(C(N)=O)c2)=O)CCC(C2CC2)(CNC(C2CCCCO2)=O)C1 C1(NC(=O)Cn2ncnn2)CN(C(c2ccc(Cl)[nH]2)=O)CC1Cc1ccccc1 Cn1cnn(CC(N2CCN(Cc3nc(C(C)(C)C)cs3)CC2)=O)c1=O C1(CC(=O)NC)CN(C(c2cncnc2)=O)CCN1C(c1cnc(C2CC2)[nH]1)=O CN1CC2(CCN(C(C3CCN(C(c4cccc(Br)c4O)=O)CC3O)=O)CC2)C1 Cc1cnccc1C=CC(=O)NC1(CF)CCN(C(=O)C(C)CO)C1 c1(C(N2CCC(NC(c3c(C)sc(Cl)n3)=O)C23CC3)=O)cncc2c[nH]nc12 N1(C(Cc2c(C)n[nH]c2)=O)CCC(c2cn(CCOC(C)C)nn2)CC1 Cc1ccc(C=CC(=O)NC2CCCC2CNC(c2nnsc2C)=O)s1 c1(C(=O)NCC2C(NC(c3ncncc3Cl)=O)CCCC2)cc(F)ccc1O C(N=c1[nH]c(N2CCc3c(nnn3C)C2)nc2c1CSC2)C1OCC(C)C1 c1(SC)ccc(CCC(=O)N(C(c2nc(C(F)(F)F)cs2)C)C2CC2)cn1 C1(C(=O)NC2(C)CN(C(C(COC)N(C)C)=O)C2)CCCN(C)C1 N1(C(C(C)NC(C)=O)=O)CCC2CN(c3cccc(F)c3C#N)CC2CC1 C1(CC(=O)NCCN(CCC)C(c2cncc(CO)c2)=O)CCOC(C)(C)C1 c1(C(=O)NC2CCN(C(C(C3CC3)OCC)=O)CC2)ccc2[nH]cc(C#N)c2c1 C1(Cl)(C(=O)NCC(C)CN(C(=O)C(C)(C)n2ccc(C3CC3)n2)C)CC12CCC2 N1(C(=O)OC(C)(C)C)CCC(c2cccc(Cl)c2)CC1.C12(CCCCC1)C(=O)N2 C1(CNC(Cc2scc(C)n2)=O)C(C)CCN1C(c1cc(C2CC2)[nH]n1)=O N1(C(Cn2cc(C(C)O)nn2)=O)CCCC(NC(C2COCCO2)=O)C1C CCC(CC)C(C)C(=O)N1CC2(C(N3CCC(CC(F)F)C3)=O)CC1CO2 C(CN=c1nc2c(ncn2C(C)C)c(NCC2CC(NS(C)(=O)=O)C2)[nH]1)SCC c1(SCC(=O)NC2(c3ccc(Cl)c(C)c3Cl)COC2)c(C)sc2ccc(Br)cc12 C1(NC(CNC(c2ccsc2)=O)=O)CN(C(=O)C=CCOC2CC2)C2CC12 Cc1cnc(Cl)nc1N1CCOCC(NC(C2C3CCCC23)=O)C1 C1(CNC(c2occ(C)c2C)=O)CCN(C(c2n[nH]cc2C2CCC2)=O)CC1C C(=O)(CS(=O)(=O)C(C)C)N(C1CN(C(c2nc(OC)c(F)cn2)=O)CC1(C)C)C c1(C(N(CC(C)NC(c2cocn2)=O)CC)=O)cc(C(N)=O)cs1 C1(NC(c2ncccc2Oc2ccccc2)=O)CCCCN(C(=O)C=C(Cl)Cl)C1 N1(C(c2c(CC)non2)=O)CC2(CCCC2)C1C(=O)NCc1nc(C)co1 N1(C(c2cnc(OC)nc2)=O)CCc2ccccc2C1CNC(=O)CSC(F)(F)F C12CCN(C13CC3)C(C1COCC1OCC=C)C(OC)OCCN2CC.SCC.CC N1(C(c2cc(-c3ccc(C)s3)[nH]n2)=O)CC(O)C(O)CC1(C)C C(=O)(C(O)CCCNC(C1CC2CC(=O)C1O2)=O)N(CCCC(C)C)C CC1CN(C(c2cccs2)=O)CCN1C(=O)CNC(=O)Oc1ccccc1 c1(C(=O)NC2C(C)CN(C(c3cnsc3)=O)CC2C)cc(O)c2ccsc2c1 C(CC(F)(F)Cn1cc(CCC(C)O)nn1)NC(CNC(CC)=O)=O c1(CCC(=O)NC2CCN(C(C3CCCOC3)=O)CC2)cncc2ccccc12 N1(C(c2cc(OCC)n[nH]2)=O)CCCC(F)(CNC(c2snc(O)c2Cl)=O)C1 c1(-c2cc(C)cc(Nc3cc(C(=O)OC)ncn3)n2)ccc2c(c1)CNCC2 Cc1cc(O)c(NCC(O)(CN(C)C)CO)cc1C(F)(F)F CC(C)C(C)(C)CNC(=O)CCC1CCN(C(=O)CN(C)C(=O)OC)C1.C(N)=O N1(C(CC(=O)NC)=O)CCCCC(NC(=O)C(c2csc(C)n2)O)C1 N1(C(C2CCC(F)(F)C2)C)CCC(O)(C#CBr)CC1 CC(O)C(F)(F)C(=O)NCC(CNC(C1SCCCS1)=O)C(F)(F)F N1(CC)CCOCC1CC(=O)NC(CNC(c1csc(C(F)F)c1)=O)C(C)C C1(CC(=O)NCC2(C(=O)OC)CC2C)CC2(C1)CN(C(c1nnn(C)c1C)=O)C2 CCCCC(C(=O)NCC(C)NC(=O)C(C)OCCOC)C(C)C C1(CC)CN(C(=O)CN2CC=CC2)CCN1C(=O)CSCC1CCCCO1 CCCC(CCC)C(=O)Nc1ccc(C2CC2(F)F)cc1 C(CC(=O)NC(C)(CC)C1CC1)(C(C)C)NC(c1c(CC)cccc1)=O c1(C(N2C(C(=O)NC(CCSCC)CO)C(O)CC2)=O)ccc(Br)nc1F Cc1cc(C(N2CC(NC(C34CCCC(C3)OC4)=O)C(C)C2)=O)c(O)cc1F c1(C(N2CC(CCNC(C=C(CC)CC)=O)OC(C)C2)=O)cnc2ccnn2c1 N1(CC)CCC2(CC1)CC2C(=O)Nc1c(CC)ccc(I)c1 c1(N(CCCCNC(C)=O)C)nc2cccnc2c(=NCCCOC(F)F)[nH]1 C(=O)(C(C(C)C)NC(=O)Cn1nnnc1C)N1C(CCC)CCC1 Cc1ccc(CC(N2CC(OCCC3CCOC3C)C2)=O)cc1 c1(CCC(=O)NCCC(F)Cn2cc(C3(C(=O)O)CC3)nn2)ccc(CO)cc1 Cc1cnc(C(N2CC(CC(C)NC(C3(O)CC3)=O)C2)=O)c(O)c1 c1(C(=O)NC2CCC(NC(=O)C(O)C3CCCC3)CC2)c(F)ccc2occc12 N1(C(C2COCC2C(F)F)=O)CCN(C(=O)Cc2cscn2)C(CO)C1 N1(C(C2C(C(C)(F)F)C2)=O)CCC(NC(=O)Cn2nnc(C3CC3)n2)C(C)(C)C1 N1(Cc2cn(C)nn2)CC2CCC1C1CN(C(c3cc(C(F)F)nn3C)=O)CC21 C1(C)(CCC(=O)NC(C)Cn2ccnc2)CN(C(c2ccccc2)=O)C1 N1(C(C[SH](CC#C)CC)=O)CCCN(C(=O)Cc2ccccc2)C(C)C1 C12(C(N3CCC(C(=O)Nc4cncc(C#N)c4)CC3)=O)CCC(CO)(CC1)CC2 c1(CC)cnccc1-c1noc(CCc2cn(C)nn2)n1 S(=O)(=O)(c1ccc2c(c1)CCCC2)c1n(CC2C(C)c3ccccc3O2)nnn1 C1(NC(c2cc(OC)ncc2)=O)CC2CC(NC(C3(OC)CCOC3)=O)CC12 C1(C(=O)N(CC(C)NC(=O)C(F)n2cccn2)C)(OC)CCCC(C)(C)C1 c1(OCC(N2CC(CN(C(C3CCC(C)(CC)O3)=O)C)C2)=O)c(C)cccc1C c1(OCC)nc(NC(C2CCN(C(c3oc(SC)cc3C)=O)C2)C)ncc1C C(=O)(CC(O)C(Cl)(Cl)Cl)NCCCCNC(c1cc(C(=O)OC)c(C)cc1)=O c1(C(=O)NC2CCN(C(c3c(C)n(C)cn3)=O)CC2C)ccc2c(n1)OCCO2 C(=O)(C(C)C(F)(F)F)N1CCC(C(=O)NCCCP(C)(C)=O)(CC)C1 Cn1nnnc1SCC(=O)NCC(C1CCCCC1)NC(=O)Cn1ncnn1 C1(CC(=O)NOCc2nc[nH]n2)CCCN(C(=O)C#CC2CC2)C1 CC1CCCC=C1C(=O)NCCc1ocnc1NC(C1(N2CCCC2)CC1)=O C1(C)(CNC(C2CN(C(c3c(C(C)C)con3)=O)CCO2)=O)CCN(C)CC1 c1(C(=O)NCC(CC)NC(=O)CN2CCOCC2=O)cc(C2CC2)oc1C1CC1 C#CCC1CC(=O)NC2(CCC2)C(=O)N2CC(C2)O1.C(=O)(N(C)C)OC C(C(C)N=c1nc2scnc2c(NCC(=O)NOC)[nH]1)N(CCCC)C N1(C(c2cc(CC)nn2C)=O)CCC(C)(NC(=O)CC23CCCC2C3)CC1 C1(C(=O)NCC2(CCC)CC2)(CNC(c2occc2CC)=O)CC2(CC2)C1 C1(C)(NC(CC2CCCC(OC)C2)=O)CCN(C(=O)Cc2cncn2C)CC1 C1(CNC(c2c(CC)scn2)=O)CCN(C(=O)CN2CCC(C)C2)C(C)C1 C1(NC(CNC(Cc2cc(COC)no2)=O)=O)CCC12CCCC2 CC1CCN(CC(=O)NCCCN(C)CCSC2CCCC(C3CC3)O2)CC1 C1(CNC(=O)C(c2ccc(F)cc2)(F)F)CCCCN1C(=O)C(F)Cl N1(C(COc2c(C)c(F)ccc2)=O)CC2CC1CCC2NC(C1(F)CCC1)=O c1(C(N2CCC(NC(CCCNC(N)=O)=O)CC2)=O)n[nH]c2c1CCOC2 C1(NC(c2c(C)c(Cl)cnc2)=O)CC2(CCN(C(=O)C(C)n3ccnc3)CC2)C1 N1(C(c2cnc(CC(C)C)s2)=O)CCN(C(=O)C2CC2)CC1CCO C(=O)(C(O)C(C)c1ccccc1)N(CC(C)(C)NC(CC(=O)NCC)=O)C N1(C(C(C)OCC=C)=O)CC2CCC1C(NC(=O)Cn1ncc3ncccc13)C2 CCC(O)C(F)(F)C(=O)NC1CC(NC(C2(S(C)(=O)=O)CC2)=O)C1 c1(NC(C2CCN(C(C3(C(C)C)CCC3)=O)CC2O)=O)c(Cl)cc(Br)c(Cl)c1Br CC(C)CCC(C)NC(C1CCN(C(C2(C)CC(C#N)C2)=O)C1)=O CCC(C(=O)N1CCN(C(c2nn(C)cc2C(=O)OC)=O)CC1C1CC1)C(C)C c1(N(C2CNCC2F)C(c2c(OC)cccc2)=O)nc(Cl)c2c(n1)COC2 C(=O)(CC(C(F)(F)F)P(C)(C)=O)N1C(C(=O)OC)CC(n2cc(CCO)nn2)C1 C1(NC(c2nc(CC)sc2)=O)CC(C(N2CCCC(CC3CC3)C2)=O)CC1O C(=O)(CCC(C)C#N)NCC1CC(OC)CN1C(c1ncc(Cl)cc1O)=O C(=O)(C1OCCc2c(O)cccc21)NC1(CC=C)CN(C(=O)Cc2cccs2)C1 c1(C(=O)NC2CCN(OCC)CC2)ccc2cc[nH]c2n1.C12(CC1)C(=O)NC2 C1(CN(C(=O)Cc2cn[nH]c2)CC)CCN(C(c2csc(Cl)n2)=O)C1 C12(C(=O)NC3C(NC(C4(CC#C)CC4)=O)CCOC3)CCC(N=[N+]=[N-])C1C2 C1(CCCC)(C(=O)NC2(CC(=O)NC(C)CSC(F)F)CC2)CCC1 O=C(C1=NOC2(CCN(c3ncnn4ccc(Br)c34)C2)C1)N1CCC(F)CC1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(C(C)NC(COCCSC)=O)C1 C(C)(C(=O)NN(C)C(=O)OC(C)(C)C)(C(C)C)NC(c1nc2cc(Br)cnc2[nH]1)C C(=O)(CCN(OC)C(=O)CN(C(=O)C(C)C1CCC1)C)NCCC(C=C)C c1(C(=O)NC2CC(NC(c3cc(C)c(O)nc3)=O)CC2O)ccc2sccc2c1 CC(CCCNC(c1ccc(C2CC2)o1)=O)NC(=O)CC1CSCCS1 c1(OC)ccc(Cl)cc1CC(=O)NC1COCC1NC(C1(C)CC1(C)C)=O N1(C(C=CC)=O)CC2(CCCC(CNC(c3cc(-c4ccccn4)[nH]n3)=O)O2)C1 N1(C(C(CC)O)=O)CC2CCC(C1)N2C(c1ccc(Cl)cc1I)=O c1(C(N2C3CC(NC(CSCCCC)=O)C2CC3)=O)n[nH]c2c1CC(C)CC2 c1(OCCCCC)ccc(COC2CC(NC(=O)C=Cc3cncs3)C2)cn1 C1(C(=O)NCC(C)OC)CN(C(=O)C(F)OC(F)(F)F)CC(C)(C)C1 O=S(=O)(c1ccc(N2CCC(Cc3ccccc3)C2)nc1)NCCN1CCCC1 c1(OC)ccc(C(=O)NC2CN(C(c3ccc(Cl)o3)=O)CC2C(F)(F)F)cc1C CC1CC(NC(=O)CN2CSCCSC2)CCN1C(=O)Cn1cc(F)ccc1=O n1(CCC(=O)NCC2N(C(c3nc(C)n(C)c3)=O)CCCC2)cc([N+](=O)[O-])cn1 c1(CCNC(C2C(C)C2C)=O)ccc(CNC(=O)C(F)n2cccn2)cc1 N1(C(c2ccc(CC)nc2)=O)C2CCCC1CN(C(=O)CC(C)(C)C(F)F)CC2 C1(CNC(CCCCOC)=O)CN(C(C2C(C)C2C)=O)CCC1(C)C C1(C)(CNC(c2n(CCC)ncc2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)C1 C1(CC)CCN(C(=O)CCC2(NC(c3cnc(C)cn3)=O)CCCCC2)CCO1 c1(C(C)NCC2CC3CC2C2CC32)ccc([Si](C)(C)C)cc1 c1(C(N(C(C)CNC(=O)C(C)O)C)=O)ncn2cc(Br)sc12 C(=O)(CCCCF)NC(CN(C(CC(C)N(C)C)=O)C)C CCC(C)(C)C(O)C(=O)NC(C)CCN(C)C(c1ccc(=O)oc1)=O c1(NC2(c3nc(C(CC)C)on3)CCC2)coc2ccc(Cl)nc12 C(=O)(CC1=CSC2=NCCN12)N1C(C(C)(C)CNC(=O)C2=NOCC2)CCC1 C12(NC(c3ccc(CCC)cc3)=O)CCC(CC1)N(C(=O)C(C)(C(C)C)OC)C2 C1(O)(C(C)NC(=O)Cn2ncnn2)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1 c1(NC(c2csc(NC(c3ccsc3)=O)n2)=O)cccc(S(=O)(=O)O)c1 Cc1ncc2n1CC(C(=O)NC1CCCN(C(=O)CNc3ncccn3)C1)CC2 C(=O)(C(O)C(F)(F)F)NC(COCCOC)C(=O)NCC(C)(O)CCO Cc1cnc(NCC(C)C)c(S(=O)(=O)N2CCCC(C(F)(F)F)C2)c1 CC(C)CCCC(=O)NC1CCC(n2cc(C(=O)NC34CCC(C3)OC4)nn2)C1 c1(NC(=O)NC2(C)CN(C(c3ccc(NC(=O)C4CC4)s3)=O)C2)cc(F)cc(F)c1 N1(C(CCC2CCN(C(C3(CC(C)C)CCC3)=O)C2)=O)CC2CC2C2CC12 C12(NC(=O)Cc3cccc(O)c3)COC(C1)C(NC(C1CCCC13CCC3)=O)C2 N1(CN(CCCC(=C)C)C)CCN(C(c2cccc(CO)c2)=O)CC1 O=C1CCCCCCN1CC(N1CC2CCC1CN2C(=O)C(O)CC(F)F)=O C1(OC)CCN(C(C2CC(C)N2C(=O)C2=C(C)CC2)=O)C1C(C)C CCC(F)(C(=O)OC)C(=O)NCC(O)CNC(=O)CC12COC(C)(C1)C2 c1(OCOC)ccccc1C(c1nc(COC)on1)(C)C c1(C(C)(C)OC)cccc(-c2c[nH]nc2C(=O)Nc2ncccn2)c1 C1(NC(CCSC)=O)CCN(C(C)C(=O)NCc2cccnc2C)CC1 C1(CNC(C(C(C)Cc2ccccc2)O)=O)CN(c2nnc(C(N)=O)s2)CCO1 C1(Nc2cc(NCc3ccc(OC)cc3)ncn2)CCC(C)(OC2CC2)CC1 C(=O)(C(F)C(C)CNC(C1CC(=O)C1)=O)N1CCC(C)CC1 C1(C)(C(N2CC(N(C(COCc3cc(C)no3)=O)C)C(F)C2)=O)CCN(C)CC1 S(=O)(=O)(C1CC2(CCC2)C1)NC(CC)CC(C)CO N1(C(CC)=O)CCC(C2CCN(c3nc(Cl)nc(C)c3F)C2)CC1 C#CCC(C(=O)N(C)CC1(CN(C(=O)CC2CN(C)C2)CCC)CC1)C1CC1 c1(CC(=O)NC(c2nccn2C)C(C)C)nccn1C C(c1cc(C)ccc1OC)=CC(=O)NC1(CNC(C(CC)OC)=O)CCOC1 C(=O)(CC(CN(C)C)C(F)(F)F)NC1C(C)CN(C(=O)C(C)(C)Cl)CC1 C(=O)(C(CNC(=O)C(c1cnn(C)c1)O)C(C)C)N(CCC#C)C N1(C(C(CC=CC)C)=O)CCCC12CCCN(C(=O)COC(F)(F)F)C2 C(=O)(CC(C(C)C)NC(c1ccncc1)=O)NC(C#C)CCC CC1CCC2(CC2)N(C(C(=O)NC2CCCCC2)C2CCOC2)C1 CCC(C(=O)NCC)C(=O)N1CC(F)CC1C(=O)NC1(CCOC)CC1 C=CC(C)CCNC(C1CC(NC(c2nncs2)=O)C1)=O C(CCC(=O)NCc1nc(C(=O)N(C2CN(C)C2)C)co1)OC(C)C c1(C(N2C(C)CC(NC(c3nn(CC)c(C)c3)=O)C2)=O)ccc([N+](=O)[O-])o1 C1(NC(=O)CC2CCOCC2)CCN(C(C2CC2c2ccccc2)=O)CC(O)C1 c1(C(=O)NC2CC(CCNC(c3[nH]cc(C)c3)=O)C2)sc(CC(F)(F)F)nc1C Cc1cc(NC(C(C)NC(c2cnn(C)c2)=O)C(C)C)n2ncnc2n1 CCC(C(=O)N1CC(C)(C)CC1CNC(C1C2COCC12)=O)C(F)(F)F N1(C(c2ccc(OC)nc2Cl)=O)CCN(Cc2ccccc2)C(C)C1C c1(C(=O)NC2CN(C(c3c(C)cnnc3)=O)C(C)C2)ccc2c(c1)CCCCN2 c1(NCC2(C=C)CCOCC2)ccc(S(=O)(=O)N2CCOC(C)C2)cc1C#N C1(C(=O)NCCN(C(=O)Cc2cnns2)CCOC)CC=CCC1C C1(NC(CCCCCOC)=O)(CNC(C2CCC(OC)C2)=O)CCC(C)(C)CC1 CC(C)CS(=O)(=O)CC(=O)NCCCCNC(=O)C(c1cc2ccccc2o1)C C(CNC(=O)CC1C=CC(NC(=O)C(C)NC=O)C1)(C(F)(F)F)OC C(=O)(C1=CC2(CCN(C(=O)CNC(C3CC3C)=O)C2)C1)NC(CSC)(C)CO c1(C(=O)NC2CC(NCc3c(C)nccc3)C2)c[nH]c2cc(F)c(F)cc12 C(=O)(N1CC(O)CCO1)C1N(C(N)=O)CCCC1.C1CCNC1 c1(C(N2C(C(C)C)C(C(=O)N(C)CCNC(N)=O)CC2)=O)ccn2ccnc2c1 C1(NC(C(CC)OC)=O)CC2(CCC(CNC(c3ccn(CCF)n3)=O)OC2)C1 N1(C(c2n(C=C)nnc2)=O)CCN(C)CC1C(=O)NOCC(C)C c1(C(N(CCNC(C(C)SCC2CCCO2)=O)C(C)C)=O)cc(F)c(Cl)cc1F c1(C(=O)NC(CCNC(C=C2CCC(C)C2)=O)(C)C)ccnc2ccncc12 Cc1nc(C2CCN(C(=O)NCC3COCCN3C3CCCC3)CC2)[nH]c1C Cc1cncnc1C(=O)NCC1(O)CC(CNC(=O)CC2CC(O)C2(C)C)C1 C=C(C)CC(C(=O)NC1CCC(NC(=O)C(N2CCC(O)CC2)C)C1)NC(C)=O C1(OCCC(=O)NCC2N(C(C(C)CSC(F)(F)F)=O)CCC2)CCN(C)CC1 c1(CC(=O)NCC2C(NC(C(COC)(C)O)=O)CC2)cc(Cl)ccc1Cl C1(NC(C=CC)=O)CCC(CNC(c2ncoc2-c2cnn(C)c2)=O)C1 N1(C(C2(C#C)CC2)=O)C2CCC1C(C(N)=O)C2.c12ccc(cc1)OCC(=O)OC2 c1(C(=O)NC(CNC(C(C)SC)=O)(C)C2CC2)c(C2CCC2)cnn1C c1(C(C)C(=O)NCCC(C)NC(c2nncs2)=O)ccnn1C Cn1c(C(N2CCC2CNC(C2CC(CCO)C2)=O)=O)cc2c(O)cccc12 C1(C(=O)NC(C)(CNC(=O)C(COC)OC)CO)(OCC)CCCC1.CSC C1(NC(c2cn(C(C)C)nc2)=O)CCN(C(=O)COc2cccnc2)CC1 C(C)(CSC)(C(=O)NCC(c1cnc[nH]1)C)NC(CCSC)=O N1(C(c2c(OC)ccnc2)=O)CCCCC(NC(c2cn[nH]c2)=O)C1 C1(C)(C(N2CC(C(C(=O)NCC3CCSCC3)OC)C2)=O)CCCCC1 C1(C(N2CC(C)C(C)C2C)=O)CC12CCN(C(=O)Cn1ccnn1)CC2 c1(C(=O)OC)cnc(C)nc1NC(CNC(c1cc2occc2s1)=O)C1CCC1 N1(C(Cc2c(C)nc(S)s2)=O)CC2(CCCC2NC(=O)C(=O)NC2CC2)C1 c1(C(N2CCCC2C2CCCOC2)=O)nc(O)nc(O)c1F C1(C(=O)NC(c2ccccc2)CNC(C2(O)CC2)=O)C2CCCCCC12 Cc1nn(CC(=O)NCCCCCN(C(=O)CC2CCCC2C)C)c(C)c1C c1(C(=O)NCC(C)NC(=O)C(c2cccc(F)c2)O)cccc2nn[nH]c12 N1(C(C=C(C)C(C)C)=O)CCC(c2n[nH]c(CNC(c3ccncc3)=O)n2)CC1 C(CCCCC(=O)NCC(CO)C(F)(F)F)N(C)C(c1ccc(F)cc1F)=O CC(C)S(=O)(=O)CC(=O)N(C(c1ccccc1)CNC(c1cc(Cl)c(Cl)[nH]1)=O)C C12(CCCCC1)n1nnnc1S2.c1(CN)ccc(C(F)C(F)(F)F)cc1 c1(OC)c(C(=O)N(CCCN(C(=O)C(OC)OC)C)C)csc1Cl N1(CC)CCOCC1C(=O)NC(C(=O)NCc1cc(C(C)C)no1)C1CCC1 CCC(O)C(C)(C)C(=O)N1CCC(C(=O)NCC2(CO)CC23CCC3)O1 O(NC(=O)C(CCF)NC(=O)CNC(C1CC1C)=O)CCC=C C1(C(=O)OCc2c(OCC)cc(C)nc2)CC(C)CC(C)C1 c1(C(C(N2C(C(C)NC(CCCOCC)=O)CCC2)=O)OC)c(F)cccc1F c1(C(N2CC(NC(c3cn(CC)nc3C)=O)CC2(C)C)=O)sc2nccn2c1C Cc1nc(C#N)cc(=NCC2CCCCN(C(c3cccc(O)n3)=O)C2)[nH]1 C12(OC)CCN(C1)C2=O.C1(C(=O)NCC2C(C(=O)OC)C2)CCC(C)(C)C1 C(=O)(C(C)(CC)CO)NCC(C(C)C)NC(C=CC)=O CC1(C(N2CCOCC(CNC(C3C=CC=CC=C3)=O)C2)=O)CCNC(=O)C1 C1(CNC(C(C(C)C)N(C)C)=O)CC2CCC(C1)N2C(=O)CCCC(=O)N(C)C C(=O)(CCCCC(=O)N1CCN(CC(=O)NC2CCC(=O)NC2)CC1)OC C1(C(=O)NCC=CCNC(=O)CC2CCSCC2)CCc2nc[nH]c2C1 [N-]=[N+]=NC1CCCN(C(=O)OC(C)(C)C)CC1.C12(CC=CC1)CCC(=O)N2 C12(C(=O)NCCOCCNC(COCC(C)C)=O)CCCC1C2Br c1(C(C)C)ccccc1C(=O)NC(C)C(C)(C)NC(=O)C=Cc1ccnn1C C=C1CCN(C(c2cn(C)c(=O)cn2)=O)C(C(N2CCC(CC3CC3)CC2)=O)C1 N(C1CCCc2cc(O)ccc21)C(CCCNS(N(CC)CC)(=O)=O)=O c1(CNC(CN(CC#C)C(c2cc(O)n(CC)n2)=O)=O)cccc(F)c1C C1(N(C(c2ccc(OCC)cc2)=O)CC)CCCN(C(=O)Cc2[nH]cnc2C)C1 N1(C(CSSC)=O)CCC(C(C)(C)O)C1.C1(=O)CN(C(N)=O)CCN1C1CC1 O(N(C)C(=O)CNC(=O)C(C1CCN(C(=O)CCc2nccn2C)C1)F)CC C1(C(N2CCC(C=C)(C(=O)NOCC(N)=O)C2)=O)CCC2(CCCC2)C1 C#CC1(C(=O)NC2CCCCC2CC(=O)NCCc2ccco2)CCCC1 C1(NC(c2cc(C3CCC3)[nH]n2)=O)CN(C(=O)CC2CC=CCC2)CC12CCC2 N1(C(c2cccc(OC)c2)=O)C2CCC1CC(N(C(=O)C(C)(O)C1CCC1)C)C2 c1(C(=O)NC2CCC(NC(C3CC(N4CC(O)C4)C3)=O)CC2)c[nH]cc(F)c1=O C1(CNC(C2(C(=O)NCCc3cocn3)CCC2)=O)CCCOCC1 C12(CNC(C)=O)CCCCC1N(C(c1cc(C)c(Cl)c(N)c1)=O)CCC2 c1(CN2CCN(CC#C)CC2)cnn2cc(-c3ccc(O)c(CC)c3)ccc12 c1(C(=O)NC2CC3CC(NC(C)=O)CC3C2)cnc2c(C#N)cnn2c1 C(=O)(C(C)(F)CS(C)(=O)=O)N(CCCN(C(C(C)OCCOC)=O)C)C C(c1ccccc1F)=CCC(=O)NCC1C(NC(=O)C=C2CCC2)CCCC1 N1(C(c2cc(OC)c(F)c(F)c2)=O)CCCC(N=c2ccnc(C3CCC3)[nH]2)C1 CC1(C(N2CCC(c3ncco3)C2)=O)CCCN(C(C2CNC(=O)O2)=O)C1 C1(C(=O)OCC)CCC2(CC1)CCN(C(C#N)CCc1cccc(Br)c1)CC2 C1(CC(=O)OC)COCC1n1cc(COCC2CC2)nn1.N1(CC(=O)N)CCCC1 C1(CCNC(COCCSC)=O)CC(F)(F)CN1C(=O)C(C1CCOCC1)F C1(C(N2CCC(CC(N)=O)C2)=O)COCCN(C(c2ocnc2C2CC2)=O)C1 C12(CCCCC1)CC(=O)N2.C(CC(=O)NCCO)N(C)CC C12(C(=O)O)CCCCC1(C(=O)O)CN(S(=O)(=O)c1scnc1C(F)(F)F)C2 C(=O)(CCS(C)(=O)=O)N1CCCC(CCC(=O)NC(CCSC)C)C1 C1(CNC(C(C(=O)OC)C)=O)CCN(C(C2C(NC(C)=O)CC2)=O)C12CCC2 N1(C(c2ccc(C)c(F)n2)=O)CCCC2(CCN(C(=O)Cc3nonc3C)C2)C1 C1(NC(=O)CCC2CC(NC(=O)CC3CC(C4CC4)C3)C2)CC(CO)C12CCC2 N1(C(c2ncn(C(C)C)c2)=O)CC(CNC(c2cn(C)nc2C2CC2)=O)CC1C c1(C(=O)NCCCC(C)NC(C(F)=C(C)C)=O)ccc(=O)n(C2CC2)c1 C(=O)(C(C)(C)C(=O)N(C)C)NCC(c1ccnn1C)C.C12CCC(CC1)CN2 C12(CNC(c3cccc(=O)o3)=O)CCC1CN(C(C1CCC=CCC1)=O)C2 N1(C(C(Cc2cnc[nH]2)NC(c2c(C)nns2)=O)=O)CCC(O)CC(C)(C)C1 C1(NC(=O)Cc2nc(C3CC3)cs2)C2COCC1CN(C(=O)C1=COCCC1)C2 C12(CNC(C3CCC(CNC(c4nc[nH]n4)=O)C3)=O)CCN(CC1)C2 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC2C(C1)NC(=O)CCN2C(=O)C(C)COC C(C(C(C)C)NC(c1ccnn1CC1CC1)=O)NC(C1(CCCC)CCC1)=O C1(CNC(Cc2nc(C)sc2)=O)CN(C(=O)Cc2ccc(O)nc2)CCO1 C1(NC(C(C)C2CCCO2)=O)CS(=O)(=O)C12CCN(c1nnc(C#N)s1)CC2 C1(C(N(CC(CC)NC(c2c(N)ccc(CC)c2)=O)C)=O)CCCC(F)(F)CC1 C(C)(C(=O)OC(C)(C)C)(C(=O)NCC1(NC(=O)CCSC)CCOC1)OC CCCCC(CC(=O)N1CC=CC1(C)CO)NC(=O)CC#N N1(C(CCCCN(C(C2(C(=O)OC)CC2)=O)C)=O)CCCC(F)CC1 N1(C(C=CC)=O)CCC(NC(c2cc(Cl)ccc2Br)=O)C(CO)CC1 c1(C(=O)NCC(C2CC2)NC(C(CC)=CC)=O)ccc(C)nc1N C1(OC)CC(NC(=O)CCSC(c2ccc(Cl)cc2)C)CN(C(=O)C(C)OC)C1 N1(C(c2c(C)cc(CO)o2)=O)CCOC2(CCN(C(C3(CO)CCCC3)=O)C2)C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2(O)CC2)=O)cc(F)ccc1Cl C1CN=C2NC(C)=CC(=NC3CC3O1)N2.c1(OC)cccc(C(C)C)c1 CC(C)CC(C)(O)C(=O)N(C)CC1CCN(C(=O)C=Cc2cn(C)cn2)C1 c1(CC(=O)N(CCN(C(C2CC(OC)C2)=O)CC)CC)ccccc1Cl C=CC(CC(=O)NCC1CCN1C(=O)C(OC)OC)c1ccccc1 c1(C(=O)NCC(CNC(c2c(C(=O)OC)c[nH]n2)=O)O)cc(C)cc(C)c1 Cc1nccc(Cl)c1C(N1CCC(CC(C)NC(C2CC(=C3CC3)C2)=O)CC1)=O C#Cc1cncc(C(=O)NC2CCN(C(c3ncnc(O)c3Br)=O)CC2F)c1 c1(C(N2CCCC(CNC(CCCC(N)=O)=O)C2)=O)ccc(Cl)c(Cl)c1N Nc1ccc(C(=O)NCC(CO)NC(c2ccoc2Cl)=O)cc1O N1(C(c2ccc(S(=O)(=O)NC)cc2)=O)CC(C)OC2(CCCC2)C1 c1(C(=O)NC2CN(C(c3cn(C)nc3Cl)=O)CC23CC3)cc(Cl)cc2c1CCC2 Cn1c(CCNC2CC(NC(=O)OC(C)(C)C)C23CCC3)cc2ccccc12 c1(NC(C2N(C)CCN(C(CC(=O)NCC)=O)C2)=O)cc(C)c(F)c(C)c1 C(=O)(C1=CC2(CCOC2)C1)N1CC(C)C(CNC(C2(c3cnn(C)c3)CC2)=O)C1 N1(C(Cc2[nH]n(CC(C)C)c(=O)c2)=O)CCC(C)N(C(=O)CN(C)C2CC2)CC1 C1(NC(c2ccc(OCC)nc2)=O)CC(C)CN(C(C2CC3C=CC2C3)=O)C1 C(=O)(C1COc2ccccc21)N1CCC(NC(=O)Cn2cc(Cl)cn2)(CO)C1 N1(C(CN(CCOC)C(c2ccc(OC)nc2)=O)=O)CCOC(C)(C(C)C)C1 N#Cc1c(NCCCCc2ccccc2)nnc2c1CCCC2.CC(C)C1CC1 C1(c2nc(CNC(C=C(C)C)=O)[nH]n2)CCCN(C(C2CCN(C)CC2)=O)C1 c1(C(=O)NC2CC(NC(CNS(CCCC)(=O)=O)=O)CC2O)ccc(N)cc1Cl C1(C(=O)NCC(CCNC(C2(COC)CC2(F)F)=O)O)CCC(=O)N(C(C)C)C1 N1(C(CCC#CC)=O)CCN(C(=O)C(C)Sc2nncn2C)C(CCO)C1 C=C(C)C(C)(O)C(=O)NC(CNC(c1ccc(F)cc1C1CC1)=O)C1CC1 Cc1ccc(N)c(C(N2CCCC(c3noc(C(C)C)n3)C2)=O)c1 c1(OC)cc(CNC2CC(NC(c3ncc(C)cc3C)=O)C2)ccc1OC(C)C C(C(=O)NCC1(C(N)=O)CN(C(=O)C(c2cccc(C)c2)=O)C1)(C(C)C)OCC c1(C(=O)NCC#CCNC(c2ncn(CC)c2)=O)ccn2c(C)cnc2c1 CC(CC(=O)NCC1C(C)CCN1C(c1cccn2ncnc12)=O)CC(C)(C)C N1(CC(C)C)CC(C(N2CCC(N(CCO)C(c3ccsc3)=O)C2)=O)CC1=O n1(CC)ccc(C(N2CC(CO)(NCCCCc3ccccc3)C2)=O)n1 N1(C(CC(CNC(C=CCOC)=O)C)=O)CC2CCC2(C(N)=O)C1 C(=O)(CCS(=O)(=O)CC(C)C)OCC(C(N1CCN(C(C)=O)CC1C)=O)C C(CCCC(CO)NC(=O)C(=C1CCCCC1)F)NC(c1c(NC)cnnc1)=O c1(C(=O)NCC(CNC(c2nc(C(C)OC)oc2)=O)O)cc(F)cc2c1CCC2 N1(C(c2cccc(C(C)=O)c2F)=O)CC2(CC(NC(C3CC3C(F)F)=O)CO2)C1 c1(N2CC3CC(NC(C(CC)OC)=O)C3C2)cnc2ccccc2n1 c1(C(N2CC(F)CC(NC(=O)CC3CCCO3)C2)=O)cnc2c(c1)C(=O)CCC2 N1(C(Cc2ccc(OC)cc2C)=O)CCC(NC(=O)CSC(F)F)C12CCCC2 N1(C(CCC=C(C)C)=O)CCN2C(=O)C(NC(c3cn(C4CC4)nn3)=O)CC2C1 C1(NC(C2(CCOC)CC2)=O)CCOC(C(=O)NC(C2CCCC2)CO)C1 C(=O)(CCCCCN1CCC(O)CC1)NC1CCN(C(COCCCC(C)C)=O)C1 Cn1nc(CNC(C2C3CCCOC23)=O)cc1C(=O)NCc1cscn1 c1(CN2C(C(N(CCCCC)CCOC)=O)CC2)c(Cl)cc(C)cc1Cl C1(NC(c2scc(OC)c2)=O)CCC12CCN(C(c1nccn1C)=O)CC2 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)NCC2(C)N=C(C)SC2)CC(O)C1 C=CCC(C)(C)CCNC(=O)C(Cc1ccoc1)NC(=O)C=CC(=O)NC1CC1 C1(n2cc(C(N3CC(F)(CO)C3)=O)nn2)CCCN(c2ccccn2)C1 c1(C(=O)NCCN(C(COCCC#C)=O)CCCN(C)C)cccc(C#C)c1F c1(C(N2CC3CC2CN3C(c2ccc(CO)cc2F)=O)=O)cc(CO)cc(F)c1 c1(C(=O)NC(CC=C)CNC(c2cc(N)ccc2Cl)=O)cncc(OC)c1C C1(OCCC)CCCN(C(=O)C(C)CNC(=O)CSC(F)(F)F)C1 Cc1cc(N)ccc1C(N1CCN(C(c2ccoc2C)=O)C(C2CC2)C1)=O C(C(C)(CC(C)C)NC(c1ccn(CC(F)F)n1)=O)NC(c1c(OC)nsc1)=O Cc1csc2c(C(=O)OCC(C)CC(F)(F)F)cccc12 C(=O)(CC(C)C(C)C)NCC(CCCC)NC(=O)C=CCCC(C)C C1(O)(C(C)NC(=O)C(Cl)=CCl)CCN(C(c2cc(N)ccn2)=O)C1 c1(NC(c2n[nH]cc2NC(c2c(O)cccc2O)=O)=O)nc2c(s1)CCCC2=O CC(C)C(O)C(=O)NC1(CC=CC(=O)NC(C)Cc2cc[nH]n2)CCC1 C1(NC(=O)NCCCC(=O)NC)CC(CO)CN1C(=O)CCNC(=O)OC C(=O)(C1=C(Cl)CCC1)NC1(C)CC(NC(C2CC(=O)NC(=O)N2)=O)C1 N1(C(c2ccc(OC)cc2)=O)CCC2C(CCCN2C(C2(C)CC=CCO2)=O)C1 CC(C)C(CNC(c1ccc(C2CC2)s1)=O)NC(=O)COc1cnn(C)c1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CC2C(=O)NC1CCC(F)CC1 C1(c2ccccc2)(NC(C(COC)OC)=O)CCN(C(=O)CSCC(C)C)CC1 Cc1ccc(N2CCCC(C(C)Nc3cc(Nc4cc(C)on4)ncn3)C2)nc1 C(=O)(C(F)(CNC(=O)COC1CCOCC1)C(C)C)N1C(CCOC)CCCC1 c1(N2CCC(N(C(C3C(=C)C3)=O)CCC)CC2)ncnc2ccccc12 c1(CCCC(=O)NCC(CNC(C(F)=CC)=O)O)c[nH]c2ccccc12 c1(C(=O)NC2CC(NC(c3ccccc3CCl)=O)C2)nc(Cl)sc1Cl C(=O)(CC(=O)N(CCn1cc(C2CCOC2)nn1)CC)OC c1(C(N(CCCN(C(c2cc(OC)n(C)n2)=O)C)C)=O)cc2cccc(C)c2s1 Cc1ncnc(C)c1C(N1CCC(C(=O)NC2(C3CCCO3)CC2)CC1)=O C(CCN=c1[nH]c(N2CCc3ccc(CO)cc3C2)nc2c1CCC2)OCCOC Cc1ccc(F)cc1CN(C1CCNC1=O)C(=O)NC(c1cccc(F)c1)CO CCCCC(C)CCC(=O)NC1CCC12CCN(C(=O)C(C)(C)CC(F)F)CC2 CCC(C)C(O)C(C)C(=O)NCC1(NC(c2ncoc2C)=O)CCC1 C1(CNC(C2N(C(C(C=C)O)=O)CC(O)C2)=O)CCCC2(CC2)C1 C1(CCN(C)C(C2CCC(=O)NC2)=O)CCCCN1C(c1ncn(C)n1)=O c1(C(=O)NC2CC2)ccc(I)cc1OC(F)F N1(C(C(C=C)(C)O)=O)CCC2(CCC(NC(c3[nH]nc(OC)c3Cl)=O)CC2)CC1 Cn1ccc2cccc(C(C(=O)NCC3CC3)N(C3CNC(=O)C34CC4)C)c12 Cc1ncc(C(c2ccccc2)NC(=O)Nc2c(Br)csc2C)c(C)n1 C(=O)(CC(C)C1CC1)NCCCN(C(C1CCC1)=O)CC.C1(=O)CN1 c1(CCC(=O)NCC(C)CNC(C2(N(C)C)CCC2)=O)csc(-c2cccs2)n1 C1(NC(c2ccncc2Cl)=O)CC(NC(C2(CO)CCC2)=O)C12CCC2 N1(C(C(C)OCC)=O)CCC(CC(C)NC(c2ncc(Cl)n2C)=O)CC1 N1(C(c2ccc(C)nc2C2CC2)=O)CC(NC(C2CC2C#N)=O)CC2(CCC2)C1 C(=O)(C(C)(C)n1cc(CC2CCCC2)nn1)OC.N12CC(C1)NC(=O)C2 N1(C(CC2CCCC(NC(c3c(COC)onc3)=O)C2)=O)CCC(C)(C2CC2)C1 C#CCCC(C(=O)N1CCOC(CCC)C1)NC(c1cc(CC)no1)=O Cc1cc(C(=O)NCC(c2ccccc2F)NC(c2cscn2)=O)ccc1Cl c1(C(N(C2(C(=O)NCCS(N)(=O)=O)CC2)C)=O)cc(C#N)c[nH]1 C1(F)(C(N2CCC(NC(=O)C(F)CC3CCC3)CC2)=O)CS(=O)(=O)CC12CCC2 N1(C(=O)C=C2CCCCC2)CCN(C(c2cccnc2)=O)C2CCCCC12 N1(C(C2(C)N(C(C(C)C(F)F)=O)CCC2)=O)CCN2CCOCC2C1 C(=O)(C(Cc1cccc(Cl)c1)CCCO)N1CCC(C)(NC(C2(O)CC2)=O)CC1 CC1CCCCCCN1C(C1CCCN(C(C2C(C)(C)C2(C)C)=O)CC1)=O C(=O)(CCS(=O)(=O)N(CC)CC)C(C1CCCC(C(N2CCC(O)C2)=O)C1)=O.CC C1(N)CN(C(c2[nH]ncc2Cl)=O)CC1COC.C1(C(=O)OCC)C(CC)C1(F)F C1(OC)CC(CNC(=O)C(c2cccc(C)c2)=O)N(C(c2cc(C)no2)=O)C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC(CNC(c2nc[nH]n2)=O)CC1 N1(C(C=COCC)=O)CCC(=CCNC(C2ON=C(C)C2C)=O)CC1 C(=O)(C(C)(C)C(=O)Nc1cccc(N2CCCCC(N)C2)c1)OCC C1(CC(=O)NCCN(C(CN(C(C)=O)C)=O)CCOC)CCOC1(C)C C(=O)(CCC(=O)N1CCC(OCCNC(c2cnncc2F)=O)C1)NC c1(CCC(=O)Nc2cccc(CNC(C34CC(CO3)C4)=O)c2)cncc(O)c1 C1(C)(CNC(C2=CC(C)(CC)C2)=O)CC(F)(F)CN1C(c1cscc1C(F)F)=O Cc1ccc(S(=O)(=O)NC(c2ccc(CCF)cc2)=O)s1 C(=O)(CCCC(=O)NC1CC1)NC(C(C(C)C)NC(=O)Cn1ccc(C(F)F)n1)C CC(C)CC(CC(C)C)C(=O)NCCOCCNC(=O)C(F)(F)C1(O)CCCC1 C1(C(=O)NCC(n2cc(CC(C)O)nn2)C)CSCCO1 C(C)(CN=c1nc2c(cnn2C)c(N2CCOC(F)(F)C2)[nH]1)(C1CCOCC1)OC c1(C(N(CCOC)C(C)C)=O)cc(C(=O)OC)no1.c1(C(=O)N)cn(CCCF)nn1 C(=O)(CCCOCCF)N(CC(=O)NCCCF)C(C)C N1(C(C2N(C)C(=O)CC2)=O)CCN(C(c2ccon2)=O)CC1CF N(C(=NCCC(C)F)NCC1(C)CCC(C(C)(C)C)CC1)CC(=O)NC Cc1cc(C(CC(=O)NC2CNC2)Oc2cc(Cl)ccn2)c(C)n1-c1ccccc1 N1(C(CN(C)CC)=O)CCN(C(C2C=CCCC2)=O)CC1CCO c1(C(=O)NCC2CC(NC(c3cccnn3)=O)C2)cc(Br)cc(F)c1F C1(CNC(=O)CC2CC3CC3C2)CN(C(=O)Cc2ccnc(O)c2)CC12CC2 Cn1ncc2ccc(C(N3CC(NC(c4cnc(N5CCCC5)nc4)=O)C3)=O)cc12 CC(C)CCC(=O)N1CCCCC1Cc1cn(C2COCC2SC)nn1 c1(CNC(=O)NC2(C(=O)OCC)CC2)cnn2c1OCCCC2 N1(C(CC2(CC)CCC2)=O)CCCCC(NC(c2cc3cscc3s2)=O)C1 c1(C(N2C(C)(C(C)C)CC2)=O)ccc(CNC(=O)COC2CCCCC2)cn1 N1(C(C(C)OCOC)=O)CC(O)CC1NC(=O)CC1COC(C)(C)C1 CCC(CC(F)(F)F)C(=O)NCC1(C)CCN(C(c2cccn2C(C)C)=O)C1 c1(OC)ccc(CNC2CC2C(=O)NCCn2cc([N+](=O)[O-])cn2)cc1Br N1(Cc2nc(COC)sc2)CCC2C1CCCN2C(=O)CO N1(C(C2(C(C)(C)O)CC2)=O)CCC(C)(C)C1CC(N1CCC12CCCC2)=O C=CCC(C)(C)CC(=O)N1CCOC(C(=O)NC(C)CC2CCC2)C1 CC(C)(C(=O)NC(C1CCOC1)CNC(c1cc(C2CC2)ccn1)=O)C(N)=O S(=O)(=O)(c1ccc(C)c(C)c1)N1CC(NC(c2nc(C)oc2)=O)C(C#N)C1 N1(C(c2n(CC)ncn2)=O)CC2CCC(N=c3[nH]c4ccccc4o3)C2C1 CC(O)CCCCCC(=O)NCC1CCN(C(C2CCC(C)(F)CC2)=O)CC1 c1(CCCN(C)C(C2CCC(C)(C)CO2)=O)c[nH]c2ncccc12 c1(OC)ccc(CO)cc1NC(C1CCN1S(=O)(=O)C1=CCC1)=O N1(C(C2CC(OCC)C2)=O)CCN(C(C2CN3CCN2CC3)=O)CC(C)(C)C1 CC(C(=O)NCC1(C(N2CC(C)(F)C2)=O)CC(C)(C)C1)C(F)(F)F C#CCC(C)C(=O)N1CCC(C)(CCNC(=O)CN2CC(=O)NC2=O)C1 Cc1nn(CC(F)F)cc1C(=O)NC12CC(CNC(=O)CC3(C)CC3F)(C1)C2 C1(CNC(C(C)NC=O)=O)CN(C(C2(C)CC=CCC2)=O)CC12CCC2 N1(C(=O)Cc2cnco2)CCC(C(=O)NCc2ccccc2Cl)(CF)C1 C12(NC(CCCN(C)C)=O)CCCC1N(C(c1cnc(C(F)F)cn1)=O)CCC2 c1(C(=O)NCC2C(C(N(CC)Cc3cccs3)=O)CCO2)cc(F)cnc1O CC1(C)CCC(C(=O)NC(C)(C)CNC(=O)CNC(c2ccoc2)=O)C1 c1(C(=O)NC2CC3C(NC(C(C)(C)Cl)=O)C3C2)cc2cnccc2[nH]1 c1(C(=O)NCC2N(C(C(CC)=CC)=O)CCCCC2)cnc2cnn(C)c2c1 C1(C(=O)NCC2(NC(C(=Cc3ccco3)C)=O)CCC2)CCCN(C(N)=O)C1 CCS(=O)CC(=O)NCC(C)N(C(=O)CCc1ccc(OC)cc1)C.C1C(=O)N1 c1(C(C)NCc2c(Cl)ncn2C)ncccc1C(F)F c1(OC)ccc2c(c1)OCC(C(=O)NC(C)CNC(=O)Cc1ccccc1Cl)C2 C12(CNC(c3n(CC)ncc3)=O)CC(NC(c3ccnc(C(N)=O)c3)=O)(CO1)C2 c1(C(=O)NCC(C)(C)NC(C2CCC2(F)F)=O)cccc2c1OCC(=O)N2 N1(C(c2nnc3n2CCOC3)C(=O)NC(C)C)CC(C(C)(C)C)c2ccccc21 N1(C(CCC(CC)C)=O)CCC2(CCN(C(c3cscc3S(C)(=O)=O)=O)C2)C1 c1(C(N2CCC(C(CO)NC(=O)CC3CC3)CC2)=O)cc(F)ccc1O C(=O)(CN=c1cc[nH]cc1)N1CC(CC(=O)Nc2c(C)c(F)ccc2)OCC1 Cc1cc(=NCCC#CBr)[nH]cc1S(=O)(=O)N1CCCC(C)C1C N1(C(Cc2c(C)nc(CC)nc2C)=O)CCC2(CC1)COC(=O)N2 Cc1oc(S(N)(=O)=O)cc1C(N1CC2(CCC(CNC(c3cnsn3)=O)O2)C1)=O CC1CCC(C(=O)NCC(C2CC2)NC(=O)C(c2ccc(Cl)cc2)O)CC1 Cn1c(C(N2CC(O)CC2CNC(c2cnc(S)n2C2CC2)=O)=O)cnc1O CC(C)C(C(=O)N1CCC(C)C1)NC(c1ccc(F)cc1)=O N1(C(C=CCOCCOC)=O)CCC(C)(CNC(c2nc(C(C)C)oc2C)=O)C1 CC(C)(C)CCC(=O)N1CC2(C)CC1(C(=O)NCC(=O)NC(C1CC1)C1CC1)C2 N1CCC(OC2CCN(C(c3[nH]c(=N)sc3)=O)C2)CC1.C1(C(=O)N)C2CNC(=O)C12 c1(CC)[nH]nc(Cl)c1C(=O)NC1CC1CNC(=O)CCC1C(=O)ON=C1C c1(CC)nc(Cl)nc(N2CCOC(CNC(=O)CC3C=CCCC3)C2)c1C#N c1(C(=O)NC(CNC(CC(CC)SC)=O)COC)cccc(N)c1F N1(C(c2ccc(COC)s2)=O)CCN(C(c2nnc(S)n2C)=O)C2CCCC12 C1(F)(C(N2CCC(C#N)C2)=O)CCN(Cc2cc(C(F)(F)F)cc(F)c2)CC1 C(C(O)(CO)CO)NC(COCCNC(=O)Cn1cnnc1O)=O c1(C2C(C(=O)NCC3CCC(NC(CCOCC#C)=O)C3)C2)ccc(C)cc1 c1(C(N2CC(CCC)N(C(=O)Cn3cncc3C)CC2)=O)cc(F)c(F)cc1N c1(NC(C)=O)cc(C(N2CC(CC(=O)NC3(n4ccnn4)CC3)C2)=O)n(C)n1 C1(C(N(CC(COCC)O)C)=O)CCCCC1NC(=O)CCC1CCOC1 c1(CN(C)C(C2CN(C(c3cncc(OC)n3)=O)C2)=O)cc(I)ccc1F c1(NC(C(=O)NC(CC(=O)OC)Cc2cccs2)=O)c[nH]c2ccc(Br)cc12 c1(-c2n(CCC)ccn2)ccc(C=C2CCCCC2)cc1C CC(CF)C(=O)NCC1CCN1C(c1snnc1SC1CCCC1)=O c1(OC)cccc(F)c1NC(C1CN(c2ccnc(Br)n2)CCO1)=O c1(-n2c(N3CCSCC3)nc(-c3scc(C)n3)n2)ccc(S(C)(=O)=O)cc1 c1(C(C(=O)NCCN(C(CCC(=C)Cl)=O)C2CC2)(C)C)ccc(Cl)cc1F Cn1nccc1C=CC(=O)NC1CCC(C)(CNC(=O)C=CCF)C1 N1(C(C2C(C)C2)=O)CCCCC(C2CN(C(c3occ4c3CCC4)=O)C2)C1 Cc1cnc(CNC2CCC(NC(c3cc(Cl)cnc3F)=O)C2)cc1Br c1(C(N2CC(CNC(C3CCCS3)=O)C2)=O)nn[nH]c1C(F)(F)F C=CC1(C(=O)NCC23CCC(F)(CC2)C3)CCN(C(=O)CN2CC(=O)NC2=O)C1 C#CCC(C)(CNC(C1N(C(=O)CN2CC(=O)NC2=O)CCC1(C)C)=O)CO C1(CCC)(NC(c2ccoc2Cl)=O)CCCN(C(=O)C=C(C)C2CCCCC2)C1 c1(C(N(C2CCN(C(=O)C(C)SC(C)C)C2)CC#C)=O)cccn2ccnc12 C1(N(C(=O)CNC(=O)C2CC2)C)CCC(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(N2CC(NC(C(C(C)O)N(C)C)=O)C(F)C2)=O)ccc2c(c1)C(=O)CCS2 c1(C(=O)NCCC(CCNC(CCC=CCC=C)=O)C)ccc(Cl)c(N)c1 C(CCC(C(=O)NCc1ccc(F)cn1)NC(c1ncccc1O)=O)OC C1(N(C(C2CCN(C)C2)=O)C)CCC2CN(C(C3CC4(CSC4)C3)=O)CC12 C(=O)(C(C(C)C)c1ccn(C)n1)NCCN(C(=O)C#CC1CC1)CC N1(C(c2n[nH]c(=N)[nH]2)=O)CCC(NC(c2ccc(Cl)nc2Cl)=O)C(CO)CC1 Cc1cc(-c2nc(C(C)C)nn2C2CCOC2C)c(F)c(Br)c1 c1(C(C)C)ccc(N)c(C(N2CC(NC(=O)C=Cc3ccc(Cl)s3)C(C)C2)=O)c1 c1(CN(C)C(=O)Nc2ccc(O)c(F)c2F)noc2c1CCCC2 c1(C(C)=O)c(CCC(N2CC(CNC(=O)C3CC3)C(O)C2)=O)c[nH]c1C C1(OC)CCCC(C(=O)NC2(C(F)F)CC(NC(=O)CC=C(Cl)Cl)C2)C1 c1(C(=O)NC(CN(C(=O)CC2CC(OC)C2)CC)C)cc(C)c(C)o1 c1(NC(=O)C=Cc2ccc[nH]2)cc(O)nn1-c1ccccc1Br c1(C(N2C(CNC(CC(CC)CC)=O)CC2)=O)cc(Br)c2ncccc2c1 c1(C(=O)NCCCN(C(C(CC)=CCCC)=O)C)snc(O)c1Cl CC1OC2(CNCC3CN(C4CCCCC4)C3)CC1(NC(C1CC1[N+](=O)[O-])=O)C2 c1(CC(=O)NCC2CN(C(COc3cc(C)on3)=O)CC2O)ncc(F)cc1F c1(C(N(CCNC(=O)CN2CCCCC2)C2CC2)=O)cc2cc(Br)sc2[nH]1 c1(C(=O)NC(CN(C(=O)CC2(OC)CC2)CC)C)cnc(OC)cn1 C#Cc1ccc(C(=O)NCCC2CCC(NC(=O)C=C3CCCCC3)C2)cc1 N1(C(C(CC)NC(=O)CSC(F)F)=O)CC(OC)C2(CC2)C1 C(=O)(C(N)CCC(C)(C)C)NC C1(NC(c2cc(CO)[nH]n2)=O)CC1C1CCN(C(=O)CC2CC23CC3)CC1 CCC(C)C(CC(=O)NC(C1CCCO1)CO)NC(=O)CCN(CC)CC C1(NC(COCc2ccc(C)cc2)=O)CN(c2cc(C)ncn2)CC2(CCC2)C1 Cc1[nH]nc(C(=O)NC2CCCC2NC(c2ccncc2Cl)=O)c1Cl c1(OCC(=O)N(CC)Cc2ccc(C)cc2)ccc(Cl)cc1F C=CC1(C(=O)NC2CC3C=CC2C3)CCN(C(c2ccc(C)nc2)=O)CC1 N1(C(c2c(F)ccc(OC)c2)C(=O)NC2CCC2)CCOc2ccc(F)cc21 CCN(N1CCC(n2nc(C)cc2C)CC1)N1CC(OC)C(CC)C1 CC1CCN(c2nnc(-c3ccccc3)s2)CC1CNC(=O)CC(C)(F)F c1(OC)ccc(C(N2CC(C3(NC(c4cc(N)ccc4F)=O)CC3)C2)=O)cc1F c1(C(=O)NC(C)CC(C)NC(c2cc(C(C)(C)C)no2)=O)sccc1S(N)(=O)=O CC1CCN(C(=O)CC2OCCC2C)CC1CNC(c1ncc[nH]1)=O C(=O)(C1SCc2cccnc21)NCC(C)NC(C1CCCN(S(C)(=O)=O)C1)=O c1(OCC=C)ccccc1C(=O)NCCN(C(=O)C(O)C(C)OC)C(C)C c1(C(=O)NCCC2CN(C(=O)C3=CCCCO3)CCO2)cc2ccsc2c(O)n1 N(C1CN(C(=O)C2=C(Cl)CCOC2)CCc2ccccc21)C(C1C(C#N)C1)=O c1(C(=O)NCCN(C(=O)C(C(C)C)NC(=O)NC)CCC)cncc(Cl)c1 C1(C(=O)Nc2ccc(Cl)cc2)CN(C(c2ccc(F)cn2)=O)CC1C1CC1 N1(C(c2nc(CC)sc2)=O)CCC(O)(CCNC(c2ccc(Cl)[nH]2)=O)C1 C(CC(C(=O)NCCC12CC(CCO1)C2)NC(=O)CC(=O)NC1CC1)OCC c1(C(N2CCN(C(C=C(CC)C)=O)CC2CF)=O)cc2cccc(F)c2s1 N1(C(C(CC(C)C)ONC(CC(C)C(C)(F)F)=O)=O)CC2CCOC(=O)C2C1 C1(NC(CCc2c(C)n(C)nc2)=O)CN(C(=O)CC#N)CC2(CC2)C1 C(C)(CCC(=O)N1CCC(CF)(NC(=O)C(CC2CCCCC2)OC)C1)OCC c1(CC(=O)NC(C2CCN(C(C3C(C)(C)C3)=O)C2)(C)C)cc(Cl)ccc1O Cc1cc(Cl)c(C(=O)NCC(C)(C)CNC(C2(C3CCCO3)CCC2)=O)cc1F N1(C(C(C)OCCC(C)C)=O)CCCC(C2CCCN(Cc3ncnn3C)C2)C1 C1(CNC(CC(C)(C)SC)=O)CCC2CN(C(=O)CCC3CC3(C)C)CC12 C(=O)(C1=CC2CCC=CCCC12)N1CC(C)(CNC(=O)CN=S(C)(C)=O)OCC1 c1(CC)ccc(C)cc1C(=O)N(CCNC(c1nc(C)n(C)n1)=O)CC C1(CCNC(C(C(C)O)N(C)C)=O)CCN(C(C2CCC2)=O)CC1(F)F C1(CC(=O)NCCOCCC(=O)NCc2ccccc2Cl)CCCC12CC2 C(=O)(C1CCCn2cncc21)NCC1CC(F)(CNC(C2(CSC)CCC2)=O)C1 C(=O)(C(C)Cc1ccccc1)NC(C1CCN(C(C2CCCC2O)=O)C1)C C1(CNC(c2cc(OCC)no2)=O)CC2COCC2N1C(=O)CN1CC(C)C1 C(CCCC(CO)NC(c1ccccc1)=O)NC(C1N(C)C(=O)CC1)=O c1(C(=O)N(CCCNC(C2(C3CC3)CC2)=O)C2CC2)cc(C#N)ccc1F N(C1CCCOc2c(OC)cccc21)C(C=C)C1CCCC1 C(C(C)CC(=O)N1CCCCC1CCCNC(=O)CCCNC(C)=O)OC c1(NC(=O)NCC(CCCOC)C)ccc(OC)c2ccnn12 CCCCCC(O)C(=O)NC1CC2(C1)CC(NC(c1cc(F)c(F)cc1F)=O)C2 c1(N2CCC(c3scc(C)n3)C2)cc(Cl)ccc1N(C)C C1(C(=O)NCC2N(C(c3n(CC(C)C)ncc3)=O)CCS2)C2CN(C)CC12 c1(C(=O)NCC2C(NC(C(CC)(C)OC)=O)C2)cc(N)c(O)c(F)c1 c12nc(cs1)C2.n1(C(CNC(C(C)SCC)=O)C)cc(-c2ccncc2)nn1 c1(C(=O)NCCN(C(COC(CC)(C)C)=O)CCOC)ccccc1NCCO c1(NC(C(C2CCN(C(COc3cc(C)on3)=O)C2)F)=O)ccc(CO)nc1 Cc1c(C(N2CC3(CC(CNC(C4CCCC4C)=O)C3)C2)=O)cccc1F Cn1nc(C(c2nnnn2C2CCC2)NCCc2ccncc2)nc1C1CC1 CCCC(O)CC(=O)NCC(C1CCCC1)NC(c1c[nH]nc1-c1ccsc1)=O c1(CNC(CC(=O)OC)Nc2ccc(Cl)cc2)ccc(-c2csc(C)c2)c(F)c1 c1(C(N(CCC(C)NC(C(CC)c2ccccc2)=O)C)=O)ccc(CC)nc1C c1(C(N2CCN(C(C(CCC)C)=O)C(C)CC2)=O)cc2c(nc1O)CCC2 CC1CCN(C(=O)Cn2ncnn2)CC1CNC(c1csc(Br)n1)=O N1(C(CNC(=O)NC)=O)CCN(C(C2CCC3(CCC3)OC2)=O)CC(CO)C1 C(CC(C)(C)CNC(c1coc(C(C)OC)n1)=O)NC(C=CC=CC)=O N1(C(C2(C(=O)NC)CC2)=O)CCC2(CC1)CC(NC(=O)C(C)CC(C)(F)F)CO2 N1(C(C2(C(N)=O)CCC2)=O)CCCN(CCNC(C2CCC3C2C3(F)F)=O)CC1 c1(C(=O)NCC2(OC)CCN(C(=O)CC(C)O)C2)ccc(C(C)=O)c(C)c1 c1(CN2C(C(N3CCC(CO)CC3)=O)CC(O)C2)cnc2cc(Cl)ccn12 N1(C(C2(OC)CC(C)C2)=O)CCC(C)(CNC(c2ccncn2)=O)C1 N1(C(C2(C)CCCC(F)(F)C2)=O)CCC2(CCCC2NC(=O)C2=CCOC2)CC1 C12(C(N(C3CCC(NC(c4ccc(F)cc4N)=O)CC3)C)=O)CC1COC2(C)C c1(CC(=O)NCC(C)(C)OCCNC(C)=O)nccc(OC)n1.C=CC1C(=O)N1 C(C(CC(=O)NCCC(C)C)OCCO)NC(CN(CC)CC)=O C1(C(=O)NCC=CCNC(C(c2n(C)cnn2)(C)C)=O)CC(C2CC2)=NO1 Cc1cnoc1NC(=O)COC(C1(c2ccon2)COC1)=O N1(C(C(CNC(c2c(C)cccc2)=O)N(C)C)=O)C2CCC1CC(F)C2 c1(C(C)C)ccc(C(N2CC(CNC(C3CCN(C)C3=O)=O)C(O)C2)=O)c(O)n1 O=S(=O)(c1ccc(Br)cc1Cl)NC1(CO)CN(Cc2nccc3[nH]ccc23)C1 N1(C(C2CC3CCC(C2)O3)=O)CCN(C(c2sncc2Br)=O)C2COCC12 N1(C(c2c(NC)cccc2)=O)CC(C(N2CC(N3CCC3)C2)=O)CC1(C)C C1(NC(c2c(OC)cccc2)=O)CC1C1CCCN(C(c2nc(O)sc2C)=O)C1 C#Cc1ccccc1CC(=O)NC1CC(CNC(C23CC(C2)C3)=O)C(O)C1 O=C1CCC2(CCCN(c3cc(N4CCNCCC4)ncn3)C2)CN1 c1(C(N2CC(NC(C3(CF)CC3)=O)CC(OC)C2)=O)coc2c(F)cccc12 N1(C(C2CN(C(C)C)C2)=O)CCC(C(C)(O)CNC(C2(C)CCOC2)=O)CC1 c1(C(=O)NCC(CCC)NC(=O)CCC2NC(=O)NC2=O)cnc2ccsc2c1 N1(C(COCC=C)=O)CCCCC(CNC(C23CCCC(CO2)C3)=O)C1 CCCCC(C(=O)NC1CN(C(c2cc(OC)n[nH]2)=O)CCC12CCC2)C(C)C N1(C(Cc2c(C)ccc(C)c2)=O)CC2CCC1C(NC(C1CN(C)C1)=O)C2 CC(C1=NOC2CCCC12)NC1CCCN(S(C)(=O)=O)C1 C1(CC)CN(C(=O)CCCn2ccnc2)CCC1NC(=O)C(c1cccnc1)O c1(C(=O)NCC(C)(CO)NC(C(CC(=O)OC)C)=O)cc2ccnc(Cl)c2s1 CN1C2CCC1CC(c1nnnn1CCCNCP(C)(C)=O)(NCCCF)C2 C=CC1OCCCC1C(=O)NCC1CC2CCC1N2C(=O)CSc1cccs1 C1(N(C(c2cc(C)n(C)n2)=O)C)CN(C(C2CC2(C)C)=O)CCC1O C1(CNC(CNC(CCC)=O)=O)(CNC(c2cnc(Cl)[nH]2)=O)CCCC1 Cc1cc(C(=O)N(CCN(C)C)Cc2ccc(F)cc2)c2nccc(C)c2c1 N1(C(C(C=CC)O)=O)CCCCC(NC(c2ccc(=O)n(C(C)C)c2)=O)C1 N12CCN(CC1C)N(CC(F)(F)F)CC2=O.c12ccc(cc1)n2C(C)=O.C(C)=O.CC N1(CC(=O)NC(CNC(CCc2ccc(C(=O)OC)[nH]2)=O)C)CCCNS1(=O)=O N1(C(C2CCC(=C)CC2)=O)CC(C)(C)OCC1CNC(=O)C(C)(C)CC1CC1 C(=O)(C(C)(C(C)C)NC(=O)NC)N1CCC(CN(C(CNS(CC)(=O)=O)=O)C)C1 N1(C(Cn2ncc(C)c2)=O)CCCN(C(C23CC(C)(C2)OC3C)=O)C(C)C1 C1(C(=O)NC(COC)C(=O)N2CC(C)(NC(C)=O)C2)CC(=O)N(OC)C1 C#CCCCC(C)C(=O)N1CCC(CC(=O)Nc2cn[nH]c2)CC1 Cc1cn2ccnc(C(N3CCCC3CN(C)C(C3CCC(=O)N3C)=O)=O)c2n1 c1(NC(C2C3(CCN(C(c4cc(C)[nH]n4)=O)C3)C2)=O)ncc(I)cc1[N+](=O)[O-] CC1(C)CCCOC1CC(=O)NNC(=O)NCC(F)(F)F CCCC(C)(C(=O)OC)NC(c1ccc(OC(F)(F)F)cc1)=O c1(C(=O)NCC2(CNC(C)=O)CC2(F)F)nn(C)cc1Cl c1(C(=O)NC(CNC(COC(CC)(C)C)=O)C2CCC2)cc(N)c(OC)cc1F N1(C(CC2CN(C(CC(C)SC)=O)CC2C)=O)CCC(F)(F)CC1C C1(NC(c2ccc(CC)s2)=O)CC2CC1CN(C(=O)C=C(C)C(C)(C)C)C2 CC1CC(C(=O)N(C(CF)CF)C)CN(C(c2ncc[nH]2)=O)C1 N1(C(CN2CC(C)C2)=O)CCC(C)C(CNC(=O)Cn2cccnc2=O)C1 c1(OC)cc(OC)c(C(F)(F)F)cc1NC(C(N1CC(F)(F)CC1C#N)=O)=O N1(C(C(CSC)N(C)C)=O)CCOC2CN(C(=O)Cc3ccc(F)cc3F)CC12 C=CCC(CNC(=O)CCCC1CCC1)C(=O)NC1CC(O)C(F)C1 CC1Cc2c(Cl)cccc2C1NCc1c[nH]c(=O)c2ccnn12 c1(C(N(CC(=O)NC(c2nc(CC)on2)C)C2CC2)=O)cccc(F)c1F C(=O)(C1=C(Cl)CCCC1)NC1C(CNC(C2C(OC)CCC2)=O)CCC1 CC1CC(NC(C2C3COCC23)=O)CN(C(c2ccc(Br)cc2O)=O)C1 c1(NCCc2cc(C)no2)cc(NC(c2csc(Br)c2)C)ncn1 CC1CCN(C(=O)Cc2cnn(CN)c2F)C1C c1(CNC(C(C(C)C)OC)c2nnnn2C(C)C)ccc2nsnc2c1 C1(C(=O)NC2CC(C)N(C(=O)OCc3ccccc3)C2)CCCC12CCC2 c1(CNC(C2(C(F)F)CC(=C)C2)=O)cccc(NC(c2cc[n+]([O-])cc2)=O)c1 C#CCCCCCCC(=O)N1C(C(=O)NCCCC2(O)CC2)CCC1C(C)C C12(CNC(C3CN(C(C)=O)C3)=O)CC1CN(C(C1CCC(=O)N1)=O)C2 c1(CCOC)nn(C)c2sc(C(N3CC(NC(c4cnc(OC)s4)=O)C3)=O)cc12 CC(O)C(F)(F)C(=O)N1CCOC(CC(=O)NCCOC(F)F)C1 c1(OC)ccc(C(=O)NCCC2CSCCN2C(=O)CC(O)C(C)C)nc1Cl c1(C(=O)NC(C2CCN(C(C(CC)NC(N)=O)=O)C2)C)c(Cl)ccc(OC)c1N CC(C(=O)NCCNc1cccnc1C(F)(F)F)S(=O)(=O)C1CCOCC1 C(c1ccc(C)cc1)=CC(=O)NC(CC)C(=O)Nc1ccc(O)c(Cl)c1 C=CCCCC(=O)NCC(C)NC(=O)C(=Cc1cccn1C)F N1(C(COCCC#C)=O)C(C(N2CCC(N(C)CC)C2)=O)CCC12CC2.C1CO1 c1(NC(C)=O)ccc(C(N2CCC(O)(CCNC(=O)C(C)CF)C2)=O)c(Cl)c1 c1(C(C)=O)cc(NC(=O)C(C)C(C)NC(=O)CN2CCCC2=O)ccc1F Cc1cc(C(=O)NCCC2(O)CCN(C(=O)CC(C)F)C2)cn1C N1(C(CCc2ncn(C)c2)=O)CCCCC(NC(C2(C(C)(C)C)CCC2)=O)C1 c1(C(N(CC(C)NC(=O)C(c2ccc(F)cc2)C)CC)=O)nnc(O)nc1O N1(C(CC=CCC)=O)CCC(C(=O)NC2CC3CCCC3C2)CC1CC N1(CC(CCCC)CC)C(=O)CCN(CCS(=O)(=O)CC2CC3(C2)CC3(F)F)C1=O O=C(C(O)CCNC(=O)C(O)C1CCCC1)N1CCC2CCC12 N1(C(c2ccc(C#C)cn2)=O)CCC2CN(C(c3ccc(CO)cc3)=O)CCC12 C1(CNC(C2(SCC)CCC2)=O)CN(C(C2CC(F)C2)=O)CC(C)(C)O1 c1(N2CC(CC)SCC2)nc(N(C)Cc2cccc(O)n2)c2c(n1)c(C)nn2C C1(NC(C(CC)=O)=O)CCSC12CN(C(=O)C(F)(F)Cl)C2 c1(OC)cc(F)c(C(=O)NCCCC(C)(C)NC(=O)CC#N)cc1S(N)(=O)=O C1(NC(CC(C)(C)OC)=O)CCC2CC1CN2C(c1nc(C2CC2)oc1C)=O C1(CNC(C(C)OCCN(C)C)=O)(NC(C2CC23CCOC3)=O)CCCCC1 c1(-n2cc(C(=O)O)nn2)ccc(C(=O)Nc2cnn(C(F)F)c2)cc1.C1CCCOC1 C1(CN(C(=O)CCn2cccn2)CC)CCCN1C(=O)CC(C1CC1)C1CC1 N1(C(C(CCC)OC)=O)CCC2(C1)CN(C(=O)C(C)=C1CCCC1)C2 C1(C(N)=O)CC=CCC1NC(C12CC1CN(C(=O)NC1CCCSC1)C2)=O C(=O)(C1=C(Cl)CCCC1)NCC1CN(C(C2C(OC)C2)=O)CC(C)C1 CC1C(NC(=O)CNC(=O)C(F)(F)F)CCCN1C(c1ccnc(F)c1N)=O N1(C(COCCC(C)C)=O)CC2CC1CN2C(c1ncc(-c2ccccc2)s1)=O c1(C(N(C2CCN(C(c3c(C#N)csc3)=O)C2)CCO)=O)ccc(F)c2c1CCC2 CC(CC(=O)NC1CCOC1C(=O)N(CC(F)(F)Cl)C)N(C)C C1(CC(=O)NC2(c3ccccc3)CN(C(=O)C=CBr)C2)CC2COCC12 c1(C(N(C2CCN(C(=O)CCCn3cncn3)C2)CC)=O)sc([N+](=O)[O-])cc1Cl C1(OC)CN(C(C2(F)CC2)=O)CC1NC(c1cnn(C(C)(C)C)c1N)=O C1(CNS(CC)(=O)=O)CCCN(C(c2cc(-c3ccccc3)oc2C)=O)C1 c1(C(N2C(C)(C(N3C(C)(C(=O)NC)CC3)=O)C=CC2)=O)ccc(C)cc1O CC1CCN(CCCNC(=O)NCCN2CCC(O)CC2)CC1 n1(CC(=O)NCC(CCC)NC(c2n(CC#C)cnn2)=O)nnc2c1CCCC2 C(CS(=O)(=O)CC1CCC1)c1cn(C(C)C(=O)N(N2C(=O)CCC2=O)C)nn1 c1(C(=O)NCCN)cc(C(CS(=O)(=O)NCCN(C(=O)OC)C(C)C)=O)oc1C.OC C(c1ccncc1)=CC(=O)NC1CC1NC(c1cc(C(F)F)ncn1)=O c1(C(C)NC(Cc2cccc(OC)c2)(C)CO)ccc(Br)c(C)c1F c1(C(N2C(CC)C(CC)CC2)C(=O)NCCSC)cc(C)c(OC)c(C)c1 C#Cc1ccc(C(C(=O)Nc2ccccc2Cl)N(C)CC2CCCN(C)C2)cn1 c1(N2CCN(C(=O)Nc3cnn[nH]3)CC2)nc2cc(Cl)cc(Cl)c2o1 C1(CNCc2cncc(N(C)C)c2)CCOC12CCOCC2 C(c1ccccn1)=CC(=O)NCCCN(C(C1(C(C)(C)O)CCC1)=O)CCO.CO Cc1nn(CC(=O)NC2C3CC(NC(c4cc(Cl)ccn4)=O)CC23)c(=O)n1C Cc1ccc(F)c(C(c2nnnn2CC2CCCO2)NCc2cnccc2C)n1 Cc1cc(C(N2CC(O)(C(C)NC(=O)Cc3c(C)cccc3F)C2)=O)cc(Cl)c1 c1(OC)cccc(CN2CC(NC(c3ccncc3O)=O)C(F)C2)c1[N+](=O)[O-] C12(C(=O)NCC3CCCC(C)C3)CCC(CN(C(C3CC4(CC4)CO3)=O)C1)C2 Cc1cnc(C(=O)NC(CNC(=O)Cc2ccc(Br)cc2C)C2CC2)c(F)c1 C(CC(=O)NCCNC(c1nn(CC)cc1Br)=O)(C(C)C)OCC C1(N(C(C(c2ccccn2)NC(C(C)SCC)=O)=O)C)CCC2(CC1)CC2 CCC(C)CC(C(=O)NC1(C)CN(C(c2csnn2)=O)C1)NC(=O)OC(C)(C)C CN1CCOC2CCN(c3nc(=NCc4ncc[nH]4)[nH]c4c3SCC4)CC12 N1(C(CCOCC#C)=O)C(NC(c2ccc(F)c(F)c2F)=O)CC2CCCCC12 CCCC(CCc1ccccc1)C(=O)NC(C)(CNC(C12CCC1CC2)=O)CC Nc1ccc(F)c(F)c1C(=O)NCC(CO)NC(=O)CN(C1CCCC1)C CC1CC(C(=O)NC2CCC(OCCCC(=O)NC3CC3)CC2)CCS1 CON(C(=O)c1cccc(CNC(c2coc(C(F)F)c2)=O)c1)C1CCCC1 C1(CC)CN(C(=O)COCC2CCC2)CCN1C(c1cncc(C2CC2)c1)=O N1(C(C(COC)(C)C)=O)CCC2(CC1)CN(C(=O)C=Cc1ccsc1)CC2CO CC1(C)C(CNC(=O)CC23CCCC2C3)CCN1C(=O)CCP(C)(C)=O C(CC1=CCN(C(=O)CC2CCCC(=O)N2)CC1)NC(C1(C)CCCOC1)=O CC1(C(=O)NC2COCCC2NC(C2(O)CCC2)=O)COc2ccccc21 c1(C(N)=O)cccc(NCC(N2CC(O)(CCNC(C3OCCCO3)=O)C2)=O)c1 C1(NC(=O)C(c2ccccc2)O)CN(C(C2(c3ccno3)CC2)=O)CC1O C1(CNC(CCc2cc(C)n(C)n2)=O)CN(C(c2ccncc2Cl)=O)CC1(C)C NS(=O)(=O)N1CC(C(N2CCN(C(C3CCC34CCC4)=O)CC2)=O)C1 n1(CC(=O)NC2CN(C(C3(OCC)CCC3)=O)C2)nc2n(c1=O)CCOC2 C1(C(C)C)CN(C(c2cn(C)cn2)=O)CCN1C(C1CCS(=O)CC1)=O CCCC(CNC(=O)Cc1ccc(O)cn1)C(=O)N(CC)OC C12(C(=O)NC3C(CNC(=O)CC4CCCOCC4)CCC3)CCC(CC1)OC2 n1(CC)cnnc1CCNC(c1cc(C2CC2)[nH]n1)c1nnnn1C(C)C n1(Cc2cn(CC3N(C(C4CC(O)(CC)C4)=O)CC3)nn2)c(C)csc1=O C(c1cccc(Cl)c1)=CC(N1CCC(N(C(C2CCC(C)C2)=O)C)CC1)=O c1(C(=O)NCCNC(=O)C(=Cc2cccnc2)F)cnc2nc(O)ccc2c1 C1(O)(CNC(C(c2ccccc2)NC(c2c(C)c[nH]c2)=O)=O)CCCN(C)C1=O N1(C(COC)C)C(=O)NC(c2nc(Cl)cs2)C2=C1CC(C)CNC2=O c1(OC)ccccc1C(CNC(=O)C(C)(F)F)NC(=O)CC1C=CCC1 C(=O)(C(CNC(C1OC2CCC1C2)=O)C(C)(C)C)NCCCC=CC C1(C(C)C)CN(C(=O)C(N2CCC(COCCO)CC2)=O)CCCO1 CC(CC1CCCC1)C(=O)N(CC(C)(C)NC(C1CCCS1)=O)C C(=O)(C1COc2ccc(Cl)cc21)NCCCOCCNC(c1cc(C)oc1C)=O c1(C(N2C(CCCNC(CNC(CC)=O)=O)CCC2)=O)ccc(C(F)(F)F)nn1 C1(NC(C2CC(C)(C(=O)OC)C2)=O)CCC2CC1CN2C(=O)CC1(C(=O)OC)CC1 Cc1nc(NCC2CCCc3nccn32)cc(=NCC2CCCSCC2)[nH]1 c1(NC(CC)CN(C)C)nc(N2CCCC(OC(C)C)C2)nc2scnc12 C1(C(=O)NCCOCCNC(C(C(C)C)c2cccnc2)=O)CCC(C)C(C)C1 c1(C(=O)NC(C2CCN(C(=O)C=CC3CCCN3C)CC2)C)cnc2n1CCC2 N1(C(c2c(C)nn(C)c2C)=O)CC(C)CN(C(C23CCCN(CC2)C3)=O)CC1C c1(C(=O)NC2C3(CN(C(CSCCCC)=O)C3)SCC2)nccn2cc(C)nc12 Cc1cc(C(N2CC(C)CC2C(N2CC3COCC3C2)=O)=O)c(F)cc1Br C1(CC(=O)NC(c2nc(=O)o[nH]2)C)CCCCC1NC(c1cc(=N)[nH][nH]1)=O Cc1cc(N)c(C(=O)NC2CCN(C(=O)C=CC3CC3)C(C)C2)cc1C c1(NC(C(n2cc(CNC3CC(N(C)C(N)=O)C3)nn2)C)=O)cc(Cl)ccc1Cl C1(NC(Cc2n(C)ncc2Cl)=O)CC(NC(c2nc(Cl)cs2)=O)C12CCOCC2 C1(C(N2CC(C)(OCC(=O)N(C)CC3(OC)CCC3)C2)=O)CCC(F)(F)C1 N1(C(C2(C(CC)=O)CC2)=O)CCCC(CNC(=O)C=CCN2CCCCCC2)C1 N1(C(CC2C(C)(C)C(O)C2)=O)CC2CCCN(C(c3ccccc3)=O)C2C1 c1(OC)ccc(CO)c(C(N)=O)c1.c12cnc(OC)nc1Nc1cc-2ccn1 N1(C(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)CCCn2ccnc2C)C2CCC12 C12(CNC(C(CN(C)C)O)=O)CCC(NC(C3(O)COC3)=O)(CC1)CO2 c1(CNC(CCOC)=O)cc(C(=O)NCC2CC(C)(O)C2)n(C)n1 c1(C(=O)NCCc2cn(CCC)nn2)cc(COCCC(F)(F)F)ccn1 CCCCC(O)CC(=O)N1CCCC(N(C)C(c2cn3ccnc3cn2)=O)C1 N1(C(c2c(C)snc2)=O)CCC(NC(=O)COCCc2cccs2)C(C)(C)C1 n1(CC(N2C(CNC(COCC=C)=O)CC3CC32)=O)ncc(O)nc1=O n1(C(C)C)ccc(C(=O)NCC2CCN2C(C2COC2)=O)cc1=O C(=O)(CCCCC(F)(F)F)NC1(C2N(C(C3C(C)OCCC3)=O)CCC2)CC1 c1(C(=O)NC2CC(NC(=O)CCc3cncs3)C2)cccc(Cl)c1Br CCCCCC(C1CC1)NC(=O)CSCCC(C)C.C12CCN(C1)CC(=O)NC2 Cc1ccc(Cl)c(OC(C)C(=O)NCCC2CN(C(=O)C(C)C(C)(C)O)C2)c1 c1(C(=O)OC)cccc2c1CCN(C(=O)OCC(CC)C(C)C)C2 C1(F)(CNC(C(c2cccc(Cl)c2)C)=O)CCN(C(=O)C=CC2CCCN2C)C1 C(=O)(CCCC(=O)c1ccc(F)cc1)NC12CC(NC(C(CO)N(C)C)=O)(C1)C2 CCC1CC(=O)NC2COCC2C(=O)N2CC(C2)O1.C(=O)(N(C)C)OC Cc1ccn2ncc(C(=O)NCCOCCNC(C3C(Cl)(Cl)C34CC4)=O)c2c1 c1(C(=O)NC2CC(C)(CNC(C3CC3C#N)=O)C2)ccc(-c2ccncc2)nc1 c1(CN=C(NC(c2ncn(C)n2)COC)NC2CCCC2)ccc(O)c(F)c1 C(=O)(CCCCCNC(=O)C(C1CCCCC1)F)N1CCC(C)(C(C)C)C1 N1(C(C2CC(=C)C2)=O)CC2CC(C)N(C(c3ccoc3CC)=O)C2C1 C=CC(CC)C(=O)N(C)CCOCCN(C(=O)CCCc1cccs1)C c1(C(N(C)CCNC(c2ccnc(OCC(F)F)c2)=O)=O)cccc(C#N)c1Br C1(C(=O)NCCNC(C=C(C)I)=O)Cc2cccnc2C1 CCC(F)(F)C(=O)N1CC2CC2(CNC(=O)Cc2ccc(Cl)cc2)C1 c1(C(=O)N)ccn2c1CS(=O)(=O)CC2.C1(C(=O)N(C)C)(COC)CCCOC1 C=CC(C)(CC)C(=O)NC(C)CCCNC(=O)CNS(=O)(=O)c1cccs1 N1(C(CCC=C)=O)CCN(C(=O)CCSc2ccccn2)C(COC)C1 CC1CCC=C1C(=O)NCC1(CNC(c2n[nH]c3c2CCC3)=O)CCN(C)C1 CC1(C(N2CC(O)(c3cn(C4COCC4O)nn3)C2)=O)COC(=O)C1 N1(C(CSc2nc(C)sc2)=O)CC(CNC(=O)C(CN(C)C)NC(N)=O)C(C)C1 C1(C(C)(C)C)CCN(C(=O)C(C2CCC2)NC(=O)C=CC2CCC2)C1 C1(NC(CCCCN(C(C)C)C)=O)COCCN(C(C2CC(=O)NC2=O)=O)C1 C(=O)(CS(=O)(=O)CC(=O)NC1CCCC(NC(=O)C(C)(C)N(C)C)C1)OC N1(C(c2c(CC)non2)=O)CC2(C1)SCCC2NC(C1CC12CCCCCC2)=O C1(C(C)NC(=O)CCCOc2ccccc2)CN(C(=O)CN2CCCC2)CCO1 N1(C(C(C)SCC)=O)CCCCC1CCC(=O)N(C1(C)CN(C)C1)C c1(NC(=O)CC2CCN(OC)C2)ccc(F)c(Cl)c1.n12ncc(C(=O)OC)c1C2 C1(C(=O)NCc2cn(CC)nc2)CC2(CC(NC(C3CCSC3)=O)C2)C1 C1(CCNC(COC(C)C)=O)CCCN(C(C2(F)C3CCCC23)=O)C1 C1(NC(CN(C)Cc2cccs2)=O)CCCN1C(=O)C=CCOc1ccccc1 N(C1c2ccccc2CC1NC(C1CCCC1O)=O)C(=O)CCCCO C(CCN=C(NCC1CC2C(C1)C2(F)F)NCCc1cccs1)OC C1(OC)CC(N(C)C(C2CC(C)(NC(c3ncccc3F)=O)C2)=O)C1(C)C c1(C(=O)NCC2CCN(C(c3nncn3C3CC3)=O)C2)ccc2c(c1)CCOC2 C1(CC(=O)NCC(CC)(C)C)C(NC(C2CC2C(F)F)=O)CC1O c1(CC)cc(C(=O)NC(C2CCN(C(c3ccc(F)c(O)c3)=O)C2)C)c(C)nn1 CC(C)CCCC(=O)N1CC(NC(=O)Cc2cscc2Br)C(O)C1 C(CCCCC(=O)NCC(C(C)C)NC(=O)Cn1ccc(C)cc1=O)OC C1(CNC(C(C)=C2CC2)=O)CCC(C)CN1C(c1cc(N2CCCC2)ccn1)=O C1(C(N(C)Cc2cc(C)on2)=O)CC2(CCN1C(=O)CC1CCCSC1)CC2 C1(C(=O)OC)CN(C(C2CCC(C)(C)CN2C(C23CC(C2)C3)=O)=O)CC1C1CC1 C1(NC(c2c(C(C)C)ncnc2)=O)CC2CC1N(C(=O)C(C#N)C(C)C)C2 C1(C(N2CCOCC2)=O)CC2(CCCCC2)S1(=O)=O.N1Cc2cnn(CCO)c2C1 C(=O)(CS(=O)(=O)CCO)N1CCC(N(C(CC(CCC)O)=O)CCO)C1 C1(C(N2CCC(C)(CNC(c3c(CC)nns3)=O)C2)=O)CC2OC1C1CC21 c1(CC(=O)NCCNC(CC(C)C2CC2)=O)cccnc1OC(F)F N1(C(CC2(COCC)CC2)=O)CCCC2C1CCCN2C(c1ccnnc1C)=O CN=c1nc(C(N2CCCOC(CNC(C3CC(CC)=NO3)=O)C2)=O)cc(C)[nH]1 N1(C(CCOCC)=O)CCC(NC(c2cnn(CC(F)F)c2)=O)C(F)(F)CC1 c1(C(=O)NC23CCN(C(c4cc(C(N)=O)oc4)=O)CC2C3)ccnc2ncnn12 C=CCCCC(N=c1nc2sccc2c(NCC(CCO)C(C)(C)C)[nH]1)C1CC1 C1(NC(C2(C)CCN(C(C(CC)C)=O)C2)=O)CC2(C1)CN(C)C2 CC(C)C(C(=O)NCC(O)CNC(=O)CSCCC#N)c1ccc(Cl)cc1 C1(NC(CN2CC(C)(C)C2)=O)CC(F)CN(C(c2ccc(F)c(N)c2)=O)C1 C1(CNC(C(C)CF)=O)CCCCN(C(=O)C=Cc2cn(C)nn2)CC1 c1(NCCCC(C)NC(C(C)C2CCOC2)=O)nc(C(F)(F)F)ccc1C#N C1(OC)CC(C(N2CC3CC3(NC(=O)COCP(C)(C)=O)C2)=O)CC1OC CON1CCC(C(=O)NC2C3CCN(C(c4ccc(O)c(Cl)n4)=O)CC23)CC1 C1(NC(=O)CCNC(C2CCC2)=O)CC2CC1N(C(c1nn[nH]c1Cl)=O)C2 N1(c2ncnc(C)c2Br)CCCC2C1CCN2Cc1ccc(Cl)s1 C1(C(=O)NC2CC(OCC)C2)CCC(CNC(c2ccncc2Cl)=O)CC1 C(=O)(CCCCN(C)C)N(CCCNC(CCn1ncc(C)c1)=O)C(C)C Cc1ccc(C(=O)NCC2(C(=O)N(C)CC3(C)CCCC3)CC=CC2)cc1 c1(C(=O)NCC(N2CCN(C(C(C)C(F)F)=O)CC2)=O)ccc2c(n1)OCCO2 c1(C(N2CC(CNC(C(F)=CC)=O)CC2(C)C)=O)ccc2c(c1)NC(=O)CCS2 C1(CCC(=O)NCC2(OC)CC2)(CNC(c2coc(C)n2)=O)CCCC1 C1(NC(c2ccc(-c3ccccc3)o2)=O)CN(C(=O)C(F)CC2CCC2)CC1O CCCC(C)(O)CC(=O)N(C1(C(=O)NC2(C)CC(O)(CO)C2)CC1)C C#CC1(NC(c2ccc(CNC(c3[nH]cnc3C)=O)o2)=O)CC2CCCC12 C1(C(=O)NC(CC(=O)OCC)C)C=CCN(C(=O)CC2(O)CCOCC2)C1 C1(C(=O)NC2(CC)CCN(C(c3c(CC)c[nH]n3)=O)CC2)CCC2(CCOC2)O1 c1(C(=O)NC2(CNC(c3c(C)coc3)=O)CC3CCC2C3)cn2ccccc2n1 c1(C(=O)NCCC2(O)CN(C(COCC)=O)C2)ccc(C2CCOCC2)nc1O C1(NC(COCC=C)=O)CC2CCC1N(C(=O)COC1CC1(F)F)C2 N1(C(c2nn(CC)c(C)c2)=O)CCCC2(NC(c3ccc(=N)[nH]c3)=O)CC12 Cc1cc(-n2cc(CONC(=O)C(C)n3ccccc3=O)nn2)cnc1C S(=O)(=O)(c1cccc2cnccc12)N1C(C(=O)NCc2ccoc2)CC(O)CC1 c1(CNC(c2nnnn2Cc2ccco2)CCSC)cc[nH]c1C(C)C N1(C(C2CCC(C)(C)C2)=O)CC2CCC2(CC(=O)NC2CCOCC2O)C1 C1(C(=O)NCC(CC=C)NC(c2[nH]nc(OC)c2Cl)=O)CC2(C1)CC(F)(F)C2 c1(OC)ncc(C(N2CC3CC3(C(N3CCC(O)C3)=O)C2)=O)cc1F N1(C(C2(NC(c3c(OC)nsc3)=O)CC2(C)C)=O)CCCOC(C(C)C)C1 CP(C)(=O)c1cscc1C(N1CC(C2(NC(C3CNC(=O)N3)=O)CC2)C1)=O C1(CN(C(=O)CC2CCCC2)C)CCCN(C(C2CC2c2cncs2)=O)C1 C1(NC(C2C(COC)CC2)=O)C=CCCC1C(N1C(C(=O)OC)CC1C)=O C1(N(C(Cn2c(=O)ccc(C)c2)=O)C)CCN(C(c2cncs2)=O)CC12CC2 CC1(C)CN(C(=O)CCC2OCCO2)CC1C(=O)CCN1CCC2CC12 N1(C(CCc2ccc(=N)[nH]c2)=O)CCC2C(NC(c3cn(CCO)nn3)=O)CC12 c1(OC(C)C(=O)OCC(CNC(=O)OCCSC)O)ccc(F)cc1.C(C)(C)C CC(C(CO)NC(c1ccc(CSC(F)F)o1)=O)NC(C1CC(F)(F)C1)=O Cc1ccc(F)c(CC(=O)NCCN(C(=O)C=CS(C)=O)CC2CC2)c1 O=S(=O)(c1ccc(N2CCC(N3CCCC3)C2)c(Br)c1)NCC1CCOC1 c1(OC)ccc(CCC(=O)NCCNC(c2cc[n+]([O-])cc2)=O)c(OC)c1OC C(C(C)(O)C(C)C)NC(C1(NC(COCCCC)=O)CC(O)C1)=O c1(C(=O)N(C2CC23CCNCC3)Cc2cc(F)cc(Br)c2F)ncnc2occc12 c1(C(=O)NCC2C(NC(CC=CC=C)=O)CCC2)cnn(CC2CC2)c1Cl c1(C(=O)NCC2C(NC(C=CCOC)=O)C2)ccnn(C)c1=O NC1CC2C(C(N3CCC4CC4C3)=O)C2C1 N1(C(c2cccc(C(C)=O)c2)=O)CC2CCC1CN2C(c1nccnc1C)=O Cc1cc(F)c(C(N2CCC(NC(c3cnsc3)=O)CC(O)C2)=O)c(F)c1 Cc1nc(-c2ccc(C(=O)OCc3nn(C(C)C)nc3Br)cc2)n2c1CCC2 Cc1[nH]nc2ccc(C(=O)NCC(C)CN(C)C(C3(C)CCCCC3)=O)c(Cl)c12 N1(C(c2c(C)cc(CO)nc2)=O)CC(C)(C)CC1CNC(c1cc(Cl)cc(Cl)c1)=O CC(CC(=O)NCC1(O)CC(CNC(=O)CC2CCC3(CC2)CC3)C1)C(F)F c1(C(=O)NCC2CCC(O)CC2)n[nH]c2c1CN(C(C1(C(F)(F)F)CC1)=O)CC2 C=Cn1nccc1C(=O)NC1(C)CN(C(=O)C(C)OCC2CC2)C1 Cc1nc(CNC(=O)NC2CCN(c3ccccc3)C2)n(C)c1C C1(CNC(CCCC=C)=O)CCCN(C(C2(C)COC(=O)OC2)=O)CC1 N1(C(CCC(=C)C)=O)CCC(CNc2ncnc(O)c2Br)C(C)C1 C(CC(C(C)C)NC(=O)CCOCC(F)F)N(C(c1cnc(C)s1)=O)C C1(C(=O)NCCCC)CCCN(C(=O)C(=Cc2cccs2)C)C1 C1(NC(C(COC(C)=O)C)=O)CCC(NC(C2CS(=O)(=O)C2)=O)CC1 Cc1nc(C(=O)N(C2CC(NC(=O)CCC(=O)N3CCOCC3)C2)C)[nH]c1C N1(C(c2c(OC)scc2)=O)CC(NC(=O)CC2(C)CC2(Cl)Cl)C(F)C1 c1(C(=O)NC2CC(NC(C3N(C)CCCC3)=O)C2)cc2nccc(C(F)F)n2n1 CC(C)CC(C)(C)C(=O)NC(CNC(c1ccc2c(c1)NCC2)=O)C1CC1 N1(C(c2csc(C)c2C)C(=O)NCCCSCC)CCC(C)(C#N)CC1 Cn1c(-c2ccccc2)c(C#N)c(=O)n1C1CCOC1 Cc1cc(NC2CCCC23CN(C(c2nn(C)cc2Cl)=O)C3)ncc1[N+](=O)[O-] C1(C(N(C(C(=O)OC)C2CC2)C)=O)CCCCC1NC(C12CSCC1C2)=O C1(CS(C)(=O)=O)(C(=O)NCCN(C(=O)CSc2cn[nH]c2)CC2CC2)CC=CC1 c1(C(=O)OCC)cc(F)cnc1NC(C1CC1NC(c1cc(Br)cc(Br)c1)=O)=O CCCCCCCCSCC(=O)NC1CCN(C(=O)CCCC#N)CC1 C(CCC(N)=O)(C(=O)N(CCCNC(=O)C=CI)C1CC1)N(C)C c1(C(=O)NC(c2ncc(C)o2)C)oc(CNC(C2(n3cccc3)CC2)=O)cc1C C1(CC(=O)NCC2CCCC2C(N2CCC3(CC2)CC3)=O)Cc2ccccc2C1 c1(NC(C2SCCN(C(C(C)(C)OC)=O)C2)=O)ccc(Cl)c(C(F)(F)F)c1 N1(C(C(CC)N(C(=O)COc2cc(C)on2)C)=O)C2CCC1CC(=O)NC2 N1(CC2CCN2C(=O)OC(C)(C)C)C(=O)CN(C)C1=O.c1(OC)cccc(C(F)(F)F)c1 C(=O)(CC(C)(C)C(F)F)N1CC(NC(Cc2nc(C(C)OCC)sc2)=O)C(O)C1 c1(N(CC(CCC)C)C)ccnc(NCc2ccc(OCC#N)cc2)n1 Cc1nc(C(N2CC(CNC(=O)C=CC3CCC3)C(C)C2)=O)ccc1Br N1(C(C(CO)NC(Cc2cnc(C(C)C)s2)=O)=O)CCN2CCCC2C1 C(=O)(CCP(C)(C)=O)NC(C(CO)NC(c1c(SC)nn(C)c1)=O)C CC(C)(C)CCC(=O)NCc1cc(C(N2CCOC(CCF)C2)=O)on1 N1(C(COCCC=C)=O)CCN(C(=O)C(c2cccc(O)c2)C)CC1 C1(C(N2CC(O)(CCNC(Cn3c(C)nnn3)=O)C2)=O)CCC(=O)N1C1CC1 CC1CN(Cc2ccc(F)c(CCC#N)c2)C(C)C1C C12(CNC(C(CCC)OC)=O)CC(CO1)N(C(=O)CCCNC=O)C2 N1(C(c2c(C)cno2)=O)CCN(C(=O)C(F)(F)C2(O)CCC2)CC(C)(F)C1 Cc1ncccc1CC(=O)NC(C)C(C)NC(=O)Cn1nc(C(F)(F)F)cc1C C1(N(C(=O)C(O)CC2CC2)C)CC2CCC(C1)N2C(=O)CN1CCCC1 c1(CC(N2C(C)CC(NC(COCCCC)=O)C2)=O)c(Br)ccc(F)c1F c1(C(N2CCC(C)C2CNC(=O)C=C(Cl)Cl)=O)cc(Cl)ccc1Cl C12(c3n(-c4cc(C)cc(Br)n4)ccn3)CCC(N=c3[nH]n4cc(C)nc4s3)(CC1)C2 CN1C2CCC1CC(=CC(=O)NCC1CC1NC(c1cc(N)c(Cl)c(O)c1)=O)C2 C(=O)(C1COc2ccccc21)N1C2C(CNC(C=C(C)C(C)C)=O)C(CCC2)C1 c1(C(=O)NC2(C)CC(NC(=O)CC3CCCOC3)C2)ccc(-c2csnn2)cc1 c1(C(=O)NCC(CNC(C23CCC2CC3)=O)OC)cc(N)nc(Cl)c1 n1(CC#C)cnnc1C(N1CCC1CC(=O)NCC(C)(O)COC)=O C1(C)(CNC(CCSCCC)=O)CCCN1C(c1cnc(SC)s1)=O Cc1cc(C(=O)NCC2CCCCC2NC(c2cc[n+]([O-])cc2)=O)cc(O)c1 N1(S(c2ccc(NCC3C(C)C3)c(Br)c2)(=O)=O)CC(C)C(=O)Nc2ccccc21 c1(C(C(=O)NC(CC)Cn2cc(-c3ccc(OC)cc3)nn2)O)ccccc1C c1(NC(C2CC(OCC)CN2Cc2c(Br)cccc2Br)=O)cccc(C)c1C C1(O)(C(C)NC(=O)CC2CC2)CCN(C(C2C(c3ccccc3)C2(C)C)=O)C1 C(CCC(=O)NCCCCCN(C(=O)Cc1csnn1)C)OCCOC Cc1ccc(C(F)F)cc1C(=O)NC1CN(C(=O)Cc2cc[nH]c2)CC1O c1(C(=O)NC2C(NC(Cn3cc(C(C)O)nn3)=O)COC2)coc2ccccc12 C1(CC)CCC1(c1nnnn1C(C)(C)C)NCCc1nc(COC)no1.C1(C)CC1 C1(CC(C(=O)NCCCC(=O)N(C)C)N)CCCC(=O)N1 N1(C(CNC(=O)OCC)=O)CCC2(CCC2CNC(c2[nH]c(O)nc2C)=O)CC1 CCCC(C(=O)N1CCC1CNC(=O)CCCCOc1cc(C(C)C)on1)N(C)C N1(C(c2ccc(NC(C)=O)s2)=O)CCC(CNC(C2(C)CC2(F)F)=O)C12CC2 c1(N2C(CC)CCC2)ncc(C(N2CCC(C(F)F)CC2)=O)cc1C C1(CNC(CNC(C)=O)=O)CC2(CCN(C(=O)C(O)C(C)C)C2)CO1 C1(O)(c2cn(-c3ncccc3C3CCNC3)nn2)CC2CCC1CC2.O=CO CCC(C)CC(=O)N1CC(CN(C(=O)C(F)(F)CC2CCCO2)C)C1 Cc1ccc(C(N2CCOC(CCNC(=O)CCCC3CC3)C2)=O)c(C)n1 CN1CCCN(C(C23CCCC2CCN3C(=O)Cn2[nH]cnc2=N)=O)CCC1 c1(C(=O)NCC2COCCN(C(C(C=C)OC)=O)C2)cnn2c(C)cccc12 O=S(=O)(c1cnc(N2CCC(c3ccccn3)C2)c(Cl)c1)NC1CC1 c1(C(=O)NC2CC(C)(NC(CCC(=O)NC)=O)C2)nc(OCC)ccc1Cl c1(C(=O)NC2(c3cn(Cc4c(C)cccc4)nn3)CCC2)ccc([N+](=O)[O-])o1 C1(C(=O)NC(CC=C)CNC(c2c(C)coc2C2CC2)=O)CCOC(C)(C)C1 C1(NC(c2cc(C(F)F)cc(F)c2)=O)CN(C(=O)C2=CCCCC2)CC1C1CC1 N1(CC(=O)NC(CC)CN(C(=O)CC2(C)CC2)C)CC(=O)NC1=O c1(NC(COC(CC)CC)=O)ccc(CNC(=O)CCc2cc[nH]n2)cc1 c1(C(C2CC(=O)N2)=O)cccc(NC(c2nc(N(C(C)=O)C)sc2)=O)c1 c1(N(CCOC)CCNC(c2nnc(C3CC3)s2)=O)ccc(C#N)cc1C Cc1cc(F)sc1C(N1CC(OCC(=O)NCCC2COCCO2)C1)=O C=C(C(=O)NC1CN(Cc2cn(C)nc2-c2ccccc2)CC1C#N)C(F)(F)F c1(CCC)c(C(=O)NCC2CCCN2C(=O)CC2CC(F)(F)C2)cnn1C c1(NCCCCC=C)ncccc1S(=O)(=O)NCC=Cc1ccccc1 c1(NC(C2N(C(c3c(C)cccn3)=O)CCSC2)=O)cccc2c1OCCC2 Cc1cc(O)c(C(=O)NC(C2CN(C(=O)CCC(=O)Nc3nccs3)C2)C)nn1 N1(C(CN2CC(C)(OC)C2)=O)CCC(CNC(=O)CN2C(C)CCC2C)C(C)C1 c1(CC(N2CCCC(NC(Cn3ccc(C)n3)=O)C2)C)ccc(F)cc1F C(C(C)C(C)C(=O)NCCOCCN(C)C(c1ccncc1Br)=O)OC c1(C(N(CCN(C(C(C)NC(C2CCC2)=O)=O)C)C)=O)ccn(C2CC2)n1 CC(CN(C)C)CN=c1[nH]c(N2CCC3CCCCC3CC2)nc2ccccc12 C1(CNC(c2cnc(O)cc2O)=O)CC2(CC2)CN1C(=O)CC1CSCCS1 CC1(C)COCC(C(N2CC(NC(=O)C(c3ccc(Cl)cc3)(F)F)C(O)C2)=O)O1 C(=O)(CCC(C)(F)F)N1CCC(C(F)F)(CNC(CCC=CCC=C)=O)C1 C1(C2CCN(C(c3ccc(CCC)cc3)=O)C2)(NC(CCCCC=C)=O)CC1 c1(C(=O)NC2C(NC(=O)Cc3cc(Br)cs3)CCC2)nccn2ccnc12 C1(C#N)(C(=O)NCC2OCC(C(=O)NC(C(=O)NCC)(C)C)C2)CCOCC1 C1(NC(c2ccc(N)c(F)c2)=O)CN(C(=O)CN2CC(=O)NC2=O)CC1C1CC1 c1(C(=O)NC(CN(C(=O)C=Cc2nnc(C3CC3)o2)C)(C)C)cccc(CO)c1 C(=O)(C(C(C)(C)C)NC(=O)CC1(COC)CCC1)NC(CCC)CO N1(C(c2c(OC)cccc2)=O)CCOCCC1C(=O)NCC1(CCO)CC1 c1(-c2cnc(SC)c(F)c2)ccc2cc(C(=O)NCCc3cccs3)[nH]c2c1 N1(CC(C)(C)S(C)(=O)=O)CCC(=O)N(CC2COCC2N2CCCC2)C1=O C1(CNC(C2(COC)CC2(F)F)=O)CN(C(C2CCC2)=O)CCC12CCC2 c1(C(N2CCCCCC2)C(=O)NCC)ccccc1OC(C)C N1(C(c2n(CC)nnc2)=O)CCCC(NC(c2ccc(F)c(C)c2)=O)C1C c1(OC)ccccc1NC(=O)CCNc1nc(-c2ccccc2SC)cs1 c1(C(=O)NCCCC2(NC(c3c(N)nccn3)=O)CC2)noc2ccc(Cl)cc12 c1(-c2nc(N)on2)ccc(CCl)cc1.COCCSC c1(C(CN2CCC2CO)OCC)ccc(N2CCCC2)cc1.C1(C)CCCCC1 c1(C(=O)NCC2C(NC(CCSC)=O)CCCC2)sc(S(N)(=O)=O)cc1C C1(C)(NC(c2cc(CC)on2)=O)CCC(NC(C2CC(COC)C2)=O)CC1 c1(C(N(C2CCN(C(c3c(OCC)cccc3)=O)C2)C)=O)cc(F)cc(C)c1N c1(C(=O)NCC2(C(C)NC(C(C)=C3CCC3)=O)CC2)conc1C(C)C C1(NC(c2nc(C(=O)OC)sc2)=O)CN(C(c2sccc2N(C)C)=O)CC1C CC1CN(C(c2cc(CNC(=O)C(C)CC(C)(C)C)[nH]n2)=O)C(C)C(C)(C)O1 C(=O)(C(C)(C)C1CCOC1)NCC=CCC(=O)NCC1CN(C(C)=O)C1 C1(C)(CNC(CC=CC=C)=O)CCCN(C(=O)C(C)CC(C)C)C1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC2C(CNC(c3n(CC)ccn3)=O)C2C1 CCN(OC)C(=O)CNC(C1C=CCN(C(=O)CN2C(=O)CNC2=O)C1)=O c1(C(=O)NCCC(C)N(C(CC(COC)C)=O)C)cc2cccc(C)c2o1 c1(CCNC(=O)OC)ccc(NC(N2CCC(C(F)(F)F)C2(C)C)=O)cc1 C1(C)(CC(=O)NCCC(C)O)CCN1C(=O)CCc1cnn(C)c1 C12(CSC)CC(C(=O)NC3CCC3NC(c3cn(CCO)nn3)=O)(CO1)C2 CCCC(CC)C(=O)N1CCC(C(C)C(=O)NC(C)C(C)CC)CC1 c1(NCCCN(C)C(C2(n3cccn3)CCCC2)=O)ccc([N+](=O)[O-])c(O)n1 Cc1ccc2oc(C(N3CCCN(C(c4cc(N)c(F)cn4)=O)CC3)=O)cc2n1 C(c1ccc2c(c1)OCO2)=CC(=O)NC(C(C)NC(=O)OC(C)(C)C)C c1(C(=O)NCC2CC(C)N(C(=O)CC(F)(F)F)C2)cccc2nc(S)oc12 Cc1cn2nc(C(=O)N(C3CCN(C(C4(C)CCOC4)=O)CC3)C)cc(C)c2n1 N1(C(C(C)(C2CCC2)NC(C(CC)C)=O)=O)CCCCCCC1CC.C1C(=O)N1 N1(C(C2=NOC(C)C2)=O)CCC2(C1)CN(C(c1ccc(C(=O)CF)cc1)=O)C2 c1(C(=O)NC2C(CCC)CN(C(=O)C(C)CC)C2)cc2ccccc2cn1 c1(C(=O)OC)cc(NC(C23CCC(OC)(CC2)CC3)=O)c(O)c(F)c1 Cc1c(C(=O)NC2C3CC4C(C3)C24C(=O)N(CC(F)F)C2CC2)c[nH]c1C#N c1(NC(CCc2cccc(N(C)C)c2)=O)n[nH]c2c1CCC(C)(C)C2 c1(COC)ccc(NC(C2(NC(c3nccn3C)=O)CCC2)=O)c(C)n1 N1(C(CCC)=O)CCN(C(C2CN(Cc3ncccc3Br)CCS2)=O)CC1 C(N=c1[nH]cnc2ccsc12)C1N(C(C(C)OCc2ccccc2)=O)CCCC1 C1(C(=O)NC(CC=C)CC=C)CC(C)(C)CN1C(c1csc(C#N)c1)=O c1(OC)cc(-c2nc(C3CCC(=O)N3)n(CC3CCCO3)n2)ccn1 N1(C(c2c(COC)cc[nH]2)=O)CCN(C(=O)CN2CCNC2=O)CC1CF S(=O)(=O)(c1ccc(C(F)F)cc1Cl)N(C(CC(C)C)C(=O)NO)C N1(CC(=O)NC2CN(C(C(C)c3ccco3)=O)C2)CCCCC1C Cc1nc(C(N2CC(CO)(NC(c3nc(O)c(C)s3)=O)C2)=O)n(C)n1 N1(C(C23CC(C)C2C3)=O)CCC2C(CCN2C(=O)CSCCN(C)C)C1 C(=O)(C(C(=O)NC(C1CN(C(C2CC3(CC3)C2)=O)CCO1)C)OC)OC c1(C(N(CC(C)CNC(=O)C(C)(C)C(C)O)C)=O)ccc([N+](=O)[O-])c(Cl)c1 C#CCC(C)(C(=O)N(C)CCOC1CC1)NC(=O)C(O)CC1CCCC1 C(C)(C(C(=O)NCC1CCCS1)NC(=O)C(c1ccoc1)OC)OC c1(C(N(C(CN(C(c2ccc(C)cc2Cl)=O)C)C)C)=O)nc2sc(C)cn2c1C c1(C(=O)NCC23CC(NC(CS(N)(=O)=O)=O)(C2)C3)c(Cl)ccc(Cl)c1O C12(Nc3ncc(C(=O)NC4(CO)CCOCC4)cn3)CCN(C1)S(=O)(=O)C2 CC(C)CCCCCC(=O)NCC(C12CCC(CC1)C2)NC(=O)CC1=CCCC1 C1(C#N)(C(N(CC(F)(F)F)CC)=O)CCCOC1 C1(CNCC2(C(N(OC)C)=O)CCCC2)CC(C)(C)CCO1 Cc1cc(N)c(C)nc1C(=O)NC1CCN(C(c2ccncc2)=O)C1C N1(C(Cc2nnc(C)o2)=O)CCN(C(C2CN(C)CCN(C)C2)=O)C2COCC12 c1(CC)ccc(C(N2CC(CCNC(=O)CCOC)C(C)C2)=O)c(C(F)(F)F)c1 c1(C(=O)NC(C2CCCN2C(=O)CCC(N)=O)C)ccc2c(c1)OCCO2 C1(C(N2CCCC(CCNC(=O)CC3CC3)C2)=O)(COC)CCC(=O)N1 Cc1cc(C(=O)NCCC2CN(C(=O)C(O)C3CC3)CCO2)nn1C(C)(C)C C1(NC(CC=C(C)C)=O)CCCN(C(=O)COC2CCCC2)C1 C(=O)(C(C)(C#N)CC)N(C(CC)CNC(=O)CC1CCC1C)C C1(C(=O)NCC(C(C)C)NC(=O)CC2(Cc3ccccc3)CC2)CCS(=O)(=O)N1 c1(CNC2C(C)CN(C(c3ccoc3)=O)C2)c(F)cccc1Br N1(C(c2ccn(CC)c2C)=O)CCC(NC(=O)C(C)P(C)(C)=O)C(O)C1 c1(C(C(=O)NCCOCC)N(CCCCC(C)C)CC)cccc(C)n1 c1(C(=O)NCCC2(O)CN(C(c3n(C)nc(O)c3)=O)C2)nnc(O)cc1O C1(C(C)NC(=O)CC2(O)CCCC2)CCN(C(=O)CCCn2cncn2)C1 CCC(C)(C)C(C)CC(=O)NC1(C)CN(C(c2ccc(NCC(C)C)nc2)=O)C1 C(=O)(CC(C(F)(F)F)c1nccn1C)N1CC(NC(CN(C)CC)=O)C(C)C1 C12CCCN(C1)C(=O)CCNC(=O)C(=O)N(C)C2.c1(CC(=O)N(C)C)cnsc1 C1(CCC)CN(C(c2sccc2-n2cnnn2)=O)CCN1C(=O)C1=C(Cl)CC1 Cc1ccc(N(C)C)c(C(=O)NC2CCC(C)N(C(C3CCCS3)=O)C2)c1 N1(C(C(CC)OC)=O)CCN(C(=O)CC2OCCCO2)CC1c1cccnc1 Cc1cccc2cc(C(=O)NCCOCCNC(c3ccc([N+](=O)[O-])[nH]3)=O)oc12 CCC(F)(F)CC(=O)NCCC1(CNC(C2CC(CCO)C2)=O)CC1 N1(C(c2cc(C)no2)=O)C2CCC1C(C)C(NC(=O)CSc1nncn1C)C2 C1(NC(C=Cc2c(C)cccn2)=O)CN(C(=O)CSC(F)F)Cc2nccn2C1 C1(C(N(C2CN(C(c3ccn(CC(F)F)n3)=O)C2)C)=O)CCCC(=O)CC1 Cc1ccc(O)cc1C(=O)NCC1CN(C(=O)Cc2ccco2)CCCO1 c1(C(=O)NCCCN(C(=O)CCCN=[N+]=[N-])C)ccc2n[nH]cc2c1 Cc1cc2ncn(CC(=O)NCC(C)CNC(=O)C(=O)CCC(C)C)c2cc1F C1(CC)CCC(C(=O)NCC2(OC)CN(C(C3CC(O)C3)=O)C2)C1 N1(C(c2c(CC)csc2)=O)CC2CCC2(CC(=O)NCCc2ncon2)C1 C1(CC)CN(C(C2C3CC2N(C(=O)C(C)(C)n2cncn2)C3)=O)CCO1 N1(C(c2c(CC)scc2)=O)CCCC(CCNC(=O)C2=CC(C)(C)C2)CC1 C(=O)(C1CCCc2nncn21)N1CCOCC(CNC(c2ccc(O)cn2)=O)C1 C1(NC(CC(CC)OC)=O)CC1C1CCN(C(=O)C(O)C2CC2)CC1 C1(C(=O)OCC)CC2(CCC2)CN1C(c1ccc(OCC)c(C(F)(F)F)c1)=O CC(CC(C)(F)F)C(=O)NCC(CNC(c1cc2c[nH]cnc-2n1)=O)CO CCN(OC)C(=O)CNC(=O)C(C(C)OC)NC(=O)CC1CSCCO1 c1(NC(N2CC3C(C(=O)OCC)(CNC3)C2)=O)nc2ccc(F)cc2[nH]1 N1(CC(NNC(C(=O)Nc2ccc(C#C)cc2)=O)=O)Cc2ccc(Br)cc2C1=O C=Cc1cccc(NC(=O)CN2CCCN(Cc3ccc(Cl)c(Cl)c3)CC2)c1 N1(C(c2cnc(OC)nc2)=O)CC(NC(=O)CCN2CCCC2)C2CCCCC12 N1(C(CCC2(C)CN(C(C34CC(CO)(C3)C4)=O)C2)=O)CCCC(O)(C2CC2)C1 C1(NC(CNC(C)=O)=O)COC2(C1)CN(C(=O)CC1CCCS1(=O)=O)C2 Cc1ncc2n1CCC(C(=O)NC(CNC(=O)CC1(O)CCCCCC1)CO)C2 S(=O)(=O)(c1ccc(N(CC)Cc2ccc(OC)cc2)c(OC)c1)N c1(C(N(C(CNC(CCC(=O)NC)=O)C)C)=O)cc(C)c(F)cc1N C1(C(N2C(CN(c3ccc(C#N)nc3)C)CCC2)=O)CC2C(O)C(O)CC12 C1(C(=O)NCC2N(C(C3C(OC)CC3)=O)CCCC2)CCC12CCOCC2 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC(C)C)NC(CCNC(COC)=O)=O c1(-n2cc(-c3c(OCC(C)(C)CO)ccnc3)nn2)cc(C(F)(F)F)ccc1Cl C1(C(=O)NCC(C2CCCN2C(c2ccc(=N)[nH]c2)=O)(C)C)CC12CC(F)(F)C2 C(N=c1[nH]cnc(C)c1Br)C1CCCC(NC(C(CC)CCOC)=O)C1 N1(C(c2cc(Cl)ncc2NCc2ncc(Br)cc2F)=O)CCn2nccc2C1 c1(CC)c(C(=O)NC2CCOCC2NC(C2CC(=O)N(C(C)C)C2)=O)ccn1C Cc1nn(CCO)cc1C(=O)NCC(O)CCNC(C1(C(N)=O)CCC1)=O C1(CC)(Cc2ccc(F)cc2)CCN(C(=O)CN(C)C(C2CCC2)=O)C1 C#CC1(C(=O)NC2(C(=O)NCC(C)CO)CCC(C)(C)C2)CCCCC1 c1(C(N2C(C(=O)NC(c3ccccc3Cl)C)CCC2C)=O)ccc(Br)cc1Br Cn1c(COCC(N2CCCC(NC(=O)Cc3nn[nH]n3)C2)=O)nnc1S C1(CNC(C(C)OCCOCC)=O)CN(C(=O)CCCC2CCCC2)CCCO1 c1(NC(=O)NC(C)CC(C)(C)O)ccc(F)c(Cl)c1F c1(C(CC2CCCO2)NC(=O)C2CC2c2ccccc2)cc2ccncc2o1 C1(NC(c2c(C)snc2)=O)CN(C(=O)Cc2cncnc2O)C2(CCOCC2)C1 C(N=c1cc(C#N)nc(C)[nH]1)C1(CNC(CC2CC(CC)OCC2)=O)CCCC1 c1(OC)ccc(Br)c(CN2CC(NC(c3ocnc3C)=O)CC(C)C2)c1 C#Cc1cc(C(N2CC(O)CC2(C)C(=O)NCC2CC2Cl)=O)ccc1C C(=O)(NNC(=O)NCC(C1CCN(C(C)=O)CC1)(C)C)C1N(CC)CCC1 C1(C(N(CCC(=O)N(CCCCC=C)C)C(C)C)=O)CC2(CCC2)C1 C1(n2cc(CN(C(C)=O)C)nn2)CN(C(C2(C(F)(F)F)CCCCO2)=O)CCO1 N1(C(c2cnc(CC)s2)=O)CCC(NC(=O)CC(C(N)=O)NC(C)=O)CC1C C1(C(=O)NC(C)CCNC(c2cn(CC3CC3)nn2)=O)CN(CP(C)(C)=O)C1 c1(-c2cc(C(=O)NC(CC)CN(C)C(c3occc3F)=O)n[nH]2)ccc(C)cc1 N1(C(N)=O)CCN(C(C2CC(=O)N(C(F)F)C2)=O)CC1 C(CC(C(=O)NC1CC(CO)C(O)C1)NC(=O)C(C)C1CCC1)OCC c1(C(=O)NCC2(CNC(c3c(CC)nco3)=O)CCCC2)cncc(Cl)c1 C(C(C)(C)C#CC(=O)N1CC(OC(F)F)C1)NC(C1CN(C)C(=O)C1)=O C1(C(NOC(CC)C)=O)CCCC(C)N1C(=O)C=CCN(CC)CC C#CC1(C(=O)NC(C)CN2CCCC2=O)CN(C(=O)C2=CCCC2)C1 C1(C(N(CCCC)CC(C)C)=O)CCN(C(=O)Cc2cncc(C)c2)CC1 c1(CNC(C2(CC)CC2)=O)ccc2c(c1)CCN(C(=O)CC1NC(=O)NC1=O)C2 CC(O)C(C)(C)CNC(C1(NC(C2(n3cccn3)CC2)=O)CCCC1C)=O.C1(C)CC1 c1(CCC(=O)NC(C)CNC(c2ccsc2OC(F)F)=O)cccc(C(N)=O)c1 c1(C(=O)NC(C(C)NC(=O)C=Cc2ccsc2)(C)C)sc(Cl)cc1Cl CC1COc2ccc(C(N3CC4CCCC4(NC(C45CCCC4C5)=O)C3)=O)cc21 Cc1[nH]c(=NCc2cc(C(F)(F)F)ccc2OCCC(O)CO)sc1C(=O)O CC1CNc2c(C(=O)NC3CC3CNC(=O)C(F)=C3CCC3)cnn2C1 N1(C(CNC(=O)NC)=O)CCC(NC(=O)Cn2ncnn2)C(C)C1 c1(C(N2CC(C)(NC(C(C=C)O)=O)C2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(C2CCC(=O)O2)=O)CCOC2(CCN(C(=O)COc3cncc(Cl)n3)C2)C1 N1(CC(=O)N(c2cc(Cl)cc(Br)c2)C)C(=O)N(C)C2(CCCCC2)C1=O CC1=NS(=O)(=O)NC=C1C(=O)N1CC2(NC(=O)C(n3cc(C)cn3)C)CCC1C2 N1(C(Cn2nc(C)oc2=O)=O)CC(CNC(C2(C)COC(=O)C2)=O)CC1(C)C N1(C(c2c(OC)c(Cl)c(Cl)cc2)=O)C2CCCC1CC(=O)NC2 c1(C(N(CCCN(C)C)C(C)C)=O)nccc2nn[nH]c12.C12CCCN(C1)C2=O N1(C(c2nc(CCC)sc2)=O)CC2(C1)SCCC2NC(C1CC1C(N)=O)=O c1(CC)conc1C(C(=O)NC1CC1)N(CCN(C)C)Cc1ccccc1 c1(N(C)CC2CC(=C)C2)nc2ccc(S(=O)(=O)NC3CC=CCC3)cc2s1 Cc1ncc([N+](=O)[O-])n1CC(N1CCC(C(F)F)(CNC(=O)C(=O)C(C)C)C1)=O c1(C(=O)NCC2C(CNC(C(CC)O)=O)C2)cc(F)cc(F)c1O C(=O)(C(Cc1cc[nH]n1)NC(C1CN(C(N)=O)C1)=O)NCC(C)(O)C1CCCC1 CCS(=O)(=O)CC(=O)NC(CC1CC1)C(=O)NCc1nnnn1C c1(C(=O)NCC2CC(OC)CN2C(C2CCOC2)=O)ccc2c(c1)COCC2 Cc1nsc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCCc2cnn(C)c2)c1N C(C(=O)N(C)CCNC(=O)CCc1c(C)noc1Cl)(C(C)(C)C)NC(C)=O C(C(=O)NNc1ccccc1S(C)(=O)=O)c1cn(-c2c(CO)ccc(C)c2)nn1 N1(C(C(F)=CC)=O)CC=C(C(=O)NC2(CC3CC3)CCC2)CC1 c1(C(N2CCC(C(=O)NCC#CC(=O)OC)OCC2)=O)ccc2[nH]ccc2n1 C1(N(C(c2c(C)cnn2C)=O)C)CC2CC1N(C(=O)C(O)Cc1cn(C)cn1)C2 C1(C(=O)NCCCCCNC(c2cc[nH]c2-c2ccccc2)=O)CC(F)C(=O)N1 N#Cc1c(-c2cn(CC(=O)NCc3ncc(F)cn3)nn2)cccc1N C(=O)(C#CC1CCCO1)NC1CC(NC(Cn2ccc(C)n2)=O)C1 C#CC1C2CCC(C2)N1N1CCC(OCC(C)(C)C)CC1 N1(C(C(c2n(C)ncc2)(C)C)=O)CC(NC(=O)Cn2cnnc2)C(O)C1 C1(CSCCNC(C2(F)CC2)=O)COCCN1C(=O)CCC1CC1CC1CC1 C=CC(C)(CC)C(=O)N1CC=CC(NC(=O)C=Cc2cn(C)nn2)C1 N1(C(CCC=CCC=C)=O)CC(C(=O)N(CC(C)O)CCC)C(F)(F)C1 C1(C(C(=O)N(CC(C(C)C)C)C)C)CCN(C(=O)Cc2ccns2)CC1 C1(CC)CN(C(C2CCC(CO)CC2)=O)CCN1C(=O)CN(C1CCC1)C C1(C(=O)NC(CN(C(c2nc(CC)sc2)=O)C)C)Cc2cc(Br)ccc2O1 C1(c2n(CCCCCC)nnn2)(NCc2ccc(CC)cc2)CC(C)N(C)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)CC3(C)OCCO3)C2)sn1 C1(NC(C2N(C(CC)=O)CCCC2)=O)CC2CN(C(=O)CSC(F)F)CC2C1 C1(CC(N2CCC(C3CC3)C2)=O)CN(C(c2c[nH]nc2-n2cnnn2)=O)CCO1 N1(CC)CC(C)N(C(=O)C#CCNC(=O)CC2OCCC2C)CC1C C(CC(C)(C)C)(C(=O)N1CC(F)(F)CC1(C)CNC(c1cocc1C)=O)OC C(C)(C(=O)N1CCCC(CNC(C2CN3CCN2CC3)=O)C1)(C(C)C)OC C1(CC(=O)NC23C(CN(C(C(C(C)C)NC(N)=O)=O)C2)C3)CCCCCCC1 N1(CCC)C(=O)NC(c2cc(Cl)cc(Cl)c2[N+](=O)[O-])C(C(=O)OCC)=C1C1CC1 CCC(C)C(C)(O)CNC(=O)C=CCN(C)C(c1cc(C#N)n(C)n1)=O c1(CC(N2C(CCNC(C3(C)CSC3)=O)CCCC2)=O)ccc2c(c1)CCC2 c1(C(N2CC(C(C)NC(c3c(C)cc(N)cc3)=O)C2)=O)cccn2c(O)nnc12 CN1CCC(C)(C(=O)NC2CCC(C)N(C(=O)C=Cc3cc[nH]n3)C2)C1=O c1(NC2C(O)COc3ccccc32)nc2ccc(Cl)cc2c(=NCC(F)(F)Cl)[nH]1 CCS(=O)(=O)c1ccc(C(=O)NC23CCC(CC2)N(C(=O)C(C)(C)F)C3)cc1 N1(C(CCCCC=CC)=O)CCC(C2CC2)C1CNC(=O)CCC1CCC1 N1(c2ncnc(=N)[nH]2)CC2CCC(NC(=O)C=CC(N)=O)CC2C1 c1(NC(=O)NC2CC(N(C)C)C2)ccc([N+](=O)[O-])c(-c2cccnc2)c1 C=CC(C)CC(=O)NCc1cncc(C(=O)NCc2cc(C(C)C)n[nH]2)c1 Cc1ccc(O)c(C(=O)NC2CCN(C(c3c(C)nn(CCO)c3C)=O)C2)n1 c1(C(N2C(CN(C(=O)C(F)OC(F)(F)F)C3CC3)CCC2)=O)nc2ccccc2[nH]1 Cc1ccn(C(C)C(=O)NC2(C(N3CC(C4CC(O)C4)C3)=O)CC(F)C2)n1 CN1C(=O)CCC1C(=O)NCC1CCCC1NC(c1ocnc1C1CC1)=O c1(C(=O)NC2C(NC(=O)CCCn3cncn3)COC2)cnccc1Cl N1(C(CCCCCOC)=O)CCN(C(c2ncc(C#N)cc2Cl)=O)CC12CCC2 C1(C(=O)OC)CN(C(C2CCCC(NC(=O)CSC)C2)=O)CCC1CO CC1(C(=O)NC(C2CCCCC2)CNC(c2nc(=N)cc[nH]2)=O)CCC(=O)N1 c1(C(CN(C)C(C2CCN(C(=O)OCC#N)C2)=O)O)ccncc1.C(C)(C)(C)O Cc1cc(Cl)c(C(C)(C)NC(=O)C(=O)N(C2CCOC2)C)cc1F CC(C)CCC(O)C(=O)N1CCC(NC(c2cncc(C(N)=O)c2)=O)CC1C C1(NC(c2nc(C)sc2C)=O)(CNC(c2nocc2C(C)C)=O)CC2CCC1C2 C=C(C(=O)N1CC(NC(C2CC(O)CCN2)=O)C(F)C1)C(F)(F)F c1(CC)cccc(CN2CC3CN(c4ccc(Cl)c(C)n4)CC32)c1[N+](=O)[O-] S(=O)(=O)(c1cc(C(N)=O)ccc1F)N1CCC(Cc2ccc(C(N)=O)cc2)C1 C12(C(N3CCC(NC(CC(C)OC)=O)(CO)C3)=O)CCC(CO)(CC1)CC2 c1(OC)ccc(C(=O)NC(CNC(C23CCCC2C3(F)F)=O)CC(C)C)c(N)c1 n1(CC)ncc2c1CCCC2N=c1[nH]c2c(c(=NCc3c(C)coc3C)[nH]1)CSC2 N1(C(CCCC#N)=O)CCC2CCN(C(c3cc4c(Cl)nccc4s3)=O)C2C1 c1(OC)ccc(C(C)NC(=O)C(n2cc(COCCO)nn2)C)cc1C CC#CC1CCN(C(=O)C(CCC)NC(c2ncc(F)cc2N)=O)C1 CCC(C)CCCCC(=O)N1CC(CN2CCN(C(=O)C(F)C(C)(C)O)CC2)C1 c1(C(=O)NCCC2N(C(CC(CC)(C)C)=O)CCSC2)cc2cc[nH]c2cn1 c1(C(=O)NCC2C(NC(c3cnc(C)[nH]3)=O)CCC2)c(C)cccc1F C1(NC(COCc2onc(C)n2)=O)CCCN(C(=O)CCC2CCC(C)O2)C1C N1(C(C2CC(NC(CC3CC(=O)NCC3)=O)C2)=O)CCCC(N=[N+]=[N-])CC1 C1(N(C(C(OC)OC)=O)C)CCC2CN(C(c3ccnc(CO)c3)=O)CC12 c1(SCCOCC(=O)N2CCC(=O)NCC2)ncccn1.CCC(C)O.CC C1(CCC)(NC(=O)C=Cc2cnc[nH]2)CCCN(C(c2cc(CC)nn2C)=O)C1 N1(C(C(N2CC(c3c(C)cccc3)OCC2)=O)=O)CC(O)C(O)CC12CCC2 C1(NC(C(N)=O)=O)CS(=O)(=O)C2CN(C(c3cccnc3O)=O)CC12 N1(C(C(CC)(C#N)CC)=O)CCC2(CC1)CN(C(=O)CC=C(Cl)Cl)CCO2 N1(C(C2(C)CCCCC2)=O)CCC2(CC1)CCN2C(c1cc2n(n1)CCSC2)=O C1(NC(C2(N(C)C)CCCC2)=O)CC2(C1)CC2NC(c1ccn(C)n1)=O c1(OCC(N2CCCC(N(CCF)C(c3cn[nH]c3)=O)C2)=O)cc(F)cc(F)c1 c1(C(=O)NCC=CCNC(CC2(C)CC2(F)Cl)=O)ccc2c(c1)C(=O)CCS2 c1(SC)nc(C)c(Cn2cc(COc3cccc(CC#N)c3)cn2)s1 C(=O)(C(C)C(O)C(C)C)N(CCC(=O)N(CCCCC#C)C)C(C)C CCCCC(C(=O)N1CCC(C)(C)C1CNC(=O)C(=O)OCC)C(C)C c1(C(=O)NCC(CNC(=O)CCC(C)N(C)C)OC)cccc[n+]1[O-] c1(C(=O)NCC(CNC(c2cc(Cl)ccc2F)=O)O)ccc(F)c(F)c1F C(=O)(C1CCCc2c(O)cccc21)NC(C)CNC(C1CCCC1C)=O S(=O)(=O)(c1ccccc1)NCCNC1C(C)CCN(C(n2c(C)ncc2)C)C1 c1(C(=O)NCCC(CNC(c2n(CC=C)ccc2)=O)OC)cc(C(C)C)n(C)n1 C(=O)(CC(C)C(C)(C)NC(c1ncncc1N)=O)N1CCC(CCOC)C1 C1(CNC(C(CC=C)C)=O)C(O)C(O)CN1C(c1nc(Cl)sc1C)=O N1(C(c2onc(C)n2)=O)Cc2nccn2CC(NC(=O)CC2CCCCC2C)C1 c1(SC)cnn(C)c1C(N1CCC(CO)(NC(=O)C=C(C)Cl)C1)=O N1(C(C(=O)C2CCCC2)=O)CC(F)(C(=O)NC(C2CCOCC2)C2CCC2)C1 C(=O)(C(C)(C)CC(F)F)N1CC2C(CNC(C3CCC(CCCC)CC3)=O)(C2)C1 c1(C(=O)NC(c2cn(CC(C(=O)OCC)O)nn2)C)cc([N+](=O)[O-])c(C)cc1C Cn1nccc1C=CC(=O)NC1(C(=O)NC2CC(O)C2(C)C)CSC1 N1(C(CC(OCC)OCC)=O)CC(NC(=O)CC(C)F)CC(C)(C)C1 c1(OCC)ccc(C(=O)NCCN(C(=O)CCSC(F)(F)F)CC)c(F)c1F C1(C(=O)NCC(CC)NC(c2cc(C)nc(O)c2)=O)CC(S(C)(=O)=O)C1 N12CCCC(CC1)CNC(=O)C(OC)C2=O.C1(C(=O)NC(C)(C)C)CCSC1 C1(NC(CC(=O)NCC(F)(F)F)=O)CC2CC(C1)N(C(c1cnc(Cl)[nH]1)=O)C2 C#Cc1ccc(C(=O)N(C2CN(C(=O)Cn3cccnc3=O)CC2F)C)cc1C c1(NCC2(C)CCOC2)ccc(S(=O)(=O)N2CCCCCC2)cc1Br C1(C2CC2)(C(=O)NCCC2CCN(C(c3nn(CC)c(C)c3)=O)CC2)CC=CC1 n1(CCC(=O)NCC2(NC(c3ccnnc3O)=O)CCOC2)ccc(O)nc1=O C1(NC(CC2CCN(C(COCCCC)=O)CC2)=O)COCC1N=[N+]=[N-] C1(NC(c2c(OC)cnc(Cl)c2)=O)CCN(C(=O)Cc2cc(C)[nH]n2)CC1(C)C c1(NC(CC)=O)cncc(C(N2CC(CNC(c3cnc(C(F)F)s3)=O)C2)=O)c1 c1(C(=O)NC(CNC(c2cccc(COC)c2)=O)COC)ccc(F)cc1F N1(C(c2n[nH]c(=N)[nH]2)=O)CC23CCCC2(C1)CN(C(=O)CC1CCOC1)C3 N1(C(=O)NCCCn2cncn2)CCOC(Cc2ccc(O)nn2)C1 C1(N(C(c2c(CC)cc[nH]2)=O)C)CN(C(=O)C(CC2CC2)OC)CC12CC2 c1(C(=O)NCC2C(C(=O)NCC(C)SC)CCC2)cn(C)ccc1=O c1(C(N2CCCCC(NC(C3C(C=C)C3)=O)C2)=O)ccc2ccsc2c1 N1(C(c2c(CC)c(OC)ccc2)=O)CC(C2CCN(C(=O)CCSC)C2)C1 Cc1oc2cc(C(N3CC(CNC(=O)Cc4ccns4)CC3C)=O)[nH]c2c1C c1(C(C(=O)NC2(CNC(C(C(CC)O)C)=O)CCC2)=O)c[nH]c2cc(F)ccc12 N1(C(CNC(CC(C)C)=O)=O)CC2CC(NC(c3cnn(C(F)(F)F)c3)=O)C1C2 c1(NC(=O)NC2CCCN(C(CCCCC)=O)C2)cc(Cl)cc(Cl)c1F Cc1ccc2oc(N3CC4CCCC(NC(C5CC(C)(F)C5)=O)C4C3)nc2c1 C1(CNC(c2cn(C(C)C)nc2)=O)CN(C(=O)CCCCNC(N)=O)CCO1 CCCCC(C(=O)NCC1(C)CCCN1C(=O)CN(c1ccccc1)C)C(C)C Cc1cc(=NCCCCCO)[nH]cc1S(=O)(=O)N(C)CC1CCCCO1 c1(C(N2CCCC(C(C)(O)CNC(C3(CF)CCC3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 C1(c2ccc(OC)cc2)COCCC1N=c1[nH]c(=N)[nH]c(Cl)c1Cl c1(C(=O)NC2CCC(N(C(CS(=O)(=O)NC)=O)C)CC2)cc2c(s1)CCCC2 c1(NC(C(C2CCC2)NC(=O)CC2C=CCC2)=O)cccc(SCCO)c1 C1(CCC)(NC(c2sccc2C(F)F)=O)CCCN(C(=O)C(C)(C)SC)C1 C(CCCC(=O)NC(CC1CC1)C1CC1)NC(C=CC(C)C)=O c1(C(=O)NCCN(C(C)C)C(C2CCCC2C2CC2)=O)cc(N(C)C)ccc1N c1(-c2c(C)cncc2)[nH][nH]c(=NC(=O)N2CCN(C)CC2C(C)C)c1C c1(C(=O)NCC2(Cn3cc(CO)nn3)CC2)c(O)ccc(Br)c1Cl O=C(CCC1CCN(C(C(C)(C)C)=O)C1)NOC1CCN(C(=O)C=CCF)CC1 N1(C(c2cnc(CC)nc2O)=O)CCC(NC(=O)C(C)(C)O)C12CCCC2 Cc1noc(C2C(C(N3CCC(NC(=O)COc4cn[nH]c4)C3)=O)C2(C)C)n1 Cc1cc(C(=O)NCC(c2ccccc2)N(C)C(C2CC(O)C2)=O)c(F)cc1Cl N1(C(c2c(C)sc(O)n2)=O)CCC(C2CC2)C1C(=O)Nc1csnc1C(C)C C(=O)(C(F)(CNC(C1CC(O)C1(C)C)=O)C(C)C)NCc1nccc(C)c1 CC1CCC(NC(=O)C=C2CCCC2)CN1C(=O)CS(=O)(=O)N1CCCCC1 N1(C(Cc2nnc(C)s2)=O)CCC(C)(CNC(c2ncc(Cl)n2C)=O)C1 N1(C(c2cc(C)no2)=O)CCC=CC1C(=O)NC(C)Cc1ccco1 c1(C(=O)NC2C(C)N(C(c3cc(CCO)on3)=O)CCC2)ccc2ccsc2c1 N1(C(C(CC)F)=O)CCN(C(c2c(C)ccnc2Cl)=O)CC(O)C1 c1(C(=O)NC(C)CCN(C(=O)C(CO)NC(N)=O)C)ccccc1-c1ncc[nH]1 C1(NC(CCCc2c(C)ccs2)=O)CCN(C(=O)CCCN(C)C)C(C)C1 C1(NC(C2(C=C)CCC2)=O)CCC2CN(C(=O)CC3CCC(=O)O3)CC2C1 c1(CNC(C2(CC)CCOC2)=O)nc(C)c(C(=O)NCCOCCN=[N+]=[N-])o1 C1(CNC(C2(CC=C)CC2)=O)CCC2(CCC2)C1NC(=O)COCC1CC1 c12ccccc1CN(C)C(=O)C2.C(=O)(C(C)CN(C)C)NCC(C1CC1)OC.O C#Cc1cncc(C(N2CCC(O)(C(C)NC(c3csc4nccn34)=O)C2)=O)c1 C1(NC(CCCCC)=O)CCN(C(=O)C(C2CC(C)(C)C2)OC)CC1O c1(-n2c(C)ncn2)ccc(NC(c2ccc(C3(C)CCO3)cc2)=O)cc1 N1(C(C(c2ccccc2C(F)(F)F)N)=O)C2CCC1C(=O)NC2 c1(N(C)C)ccc(C(=O)NCC2(O)CN(C(=O)CC3CCCOC3)C2)cn1 c1(C(=O)NC2(CNC(c3ccn(C)c3)=O)CCOC2)cc(O)nn1C c1(C(N2CC(C(=O)NC3CCC(F)(F)C3O)(COC)C2)=O)cccc2nn[nH]c12 c1(C(=O)NC2C(NC(=O)Cn3cnnc3O)CC2)ccc(C2CC2)nc1O c1(C(=O)NCCCN2CCN(C(c3n(C)ncc3Cl)=O)CC2)cc(O)cc(=O)o1 C=CC1(CC(=O)NCC2(O)CCCOC2)CN(C(=O)C(O)C2CC2)C1 C1(C(=O)NC2CC(C)(NC(c3cc(CCC)no3)=O)C2)CCS(=O)(=O)N1C C1(CC(=O)NC2CCC3(CC3)C2)CN(Cc2ccc[n+]([O-])c2)CCO1 C1(NC(C2(C)CCCO2)=O)CC2CCCC(C1)N2C(c1cc2cn[nH]c2cn1)=O c1(C(=O)NCCC(C)NC(C2(C(C)C)CCC2)=O)c(N)cc(Cl)cc1F c1(C(N2CCC(C)(NC(C(C)CC3CCCC3)=O)C2)=O)cc(=N)[nH]c(Cl)n1 C(C(C)(C)CNC(=O)C(C)N(C(c1cnccn1)=O)C1CC1)SC C(CCC(=O)O)(C(=O)O)NC(CC1N(CCS(N)(=O)=O)CCC1)=O C1(C(=O)NCC2CC(F)(CNC(C3(C(=O)NC)CCC3)=O)C2)Cc2cccnc2C1 c1(-c2nn(CCC(C)C)c(C3C(C)C3C3CC3)n2)cccc(Cl)c1 C#CCC(C)(C)CNC(=O)C(C)(C)C1CCN(C(c2cc(OC)n[nH]2)=O)C1 CS(=O)(=O)c1cc(C(=O)NC2CC(CCNC(=O)Cn3cnccc3=O)C2)cs1 C1(CC(=O)NC(C2CCCN(C(c3nc(=N)cc[nH]3)=O)C2)C)CCCNC(=O)C1 c1(-c2cnc(NC(CC(=O)OC(C)(C)C)=O)o2)c(Cl)cccc1Cl C=CC1(C(=O)NC2CC(CO)C3CC23)CCN(C(=O)C(C)N2CCCC2)C1 C1(NC(C=NOC)=O)CCN(C(c2cnc(CC3CC3)s2)=O)CC1CO N1(CC(=O)NC(CN(C(C2CC(C)C2)=O)CCO)C)OC(C)(C)CC1=O C(CC(O)CNC(c1cncn1C)=O)NC(C(C)OCC#C)=O C1(C(=O)NCC23CC(C(=O)NCC4C(OCC)C4)(OC2)C3)CCC2(CCC2)CO1 C1(N(C(CC(C)SC)=O)CCF)CCCN(C(c2nc(O)c(C)s2)=O)C1 C1(C(=O)NCC(CN(C(C(C)(C2CC2)OC)=O)C)(C)C)CN(CP(C)(C)=O)C1 N1(C(CC(COC)C)=O)CCC(NC(C2COCC(C)(C)O2)=O)C2(CCC2)C1 N1(C(C2C(COC)CC2)=O)CCC2C(NC(=O)CCCC3CCCC3)C2C1 C(=O)(C(C)(C)N=[N+]=[N-])N1C(C(=O)NCCCCCN(C)CC)CCCC1 c1(CC(=O)N(C)CC2(O)CN(C(c3ccc(O)nc3)=O)C2)ccc2c(c1)COC2 c1(C(N(CC(C)NC(=O)C(C)C2CCCC2)C)=O)c[nH]c(=NCC(F)(F)F)cn1 c1(C(N(C2CCC(NC(=O)Cn3cnc(=N)[nH]3)CC2)C)=O)ccc2cccnn12 C=CC(C)(O)CC(=O)NCC1CCCN1C(c1cccc(C)n1)=O C(=O)(C#CC1CC1)NCCOCCC(=O)NC(C1CCC1)C N1(C(CC2(CNC(C(C3CCC(O)CC3)(C)C)=O)CCCC2)=O)CC2C(CO)C2C1 c1(OC)ccc(C(F)(F)C(=O)NC2CC(NC(C3(O)CC3)=O)C2)cc1 C1(C2CCCN(C(c3ccc(Br)s3)=O)C2)(NC(=O)Cc2ccno2)CC1 N1(C(C2(C)N(C)CC(OC)C2)=O)C2CCC1CN(C(=O)CN1CC(C)(C)C1)C2 C1(C)(CNC(CNC(=O)OC)=O)CCN(C(C2(C(C)C)CNC(=O)C2)=O)C1 c1(C(=O)NC(CC(C)C)CNC(=O)CC(F)(F)C(C)C)cnc2c(ccn2C)c1 c1(C(=O)NCCN(CCOCCO)C(C2CC2F)=O)cc(F)ccc1C(F)F N1(C(CC)C)C(=O)NC(c2cc(Br)c[nH]2)C2=C1CC(C(=O)O)NC2=O C(=O)(C(CC)(CC)C(C)C)NC1C(CNC(Cc2n(CC)ncc2)=O)CC1 C1(C(=O)NC(CCC)CO)(NC(c2ccc(O)nc2)=O)CCN(C)C1 c1(C(C)NC(c2ccc(C)o2)C)ccc(NCc2cc[nH]n2)cc1 C1(NC(C2(C(=O)NCC(C)CC3CC3)CCCC2)=O)CC(F)CN(C(C)=O)C1 N1(C(c2c(OCCOC)cccc2)=O)CCC(NC(C2C(C)C2C)=O)C(F)C1 c1(SC)ccccc1.N1(CC(=O)N(CC(=O)NCC(C)N)C)CC(C)(C)C1 c1(OC)ccc(Br)c(S(=O)(=O)NC(=O)C(C(F)(F)F)N2CCNC2=O)c1 O(Nc1nccc2c(Br)c[nH]c12)C(COCC)C C(=O)(C(CO)N(C)C1CC1)N(CC(=O)NC(CC1CC1)C1CC1)CC#C c1(CC(C)C(=O)NC2CCN(C(=O)OC(C)(C)C)C23CC3)ccc(F)c(Cl)c1 N1(C(Cn2nnc(C)n2)=O)CCCC(NC(C2CCC(=O)N2)=O)CCC1 c1(C(=O)NCC(CC)(C)NC(=O)C(c2cn(C)nc2C)C)cc(C)nn1CCO c1(C(N(C2CCCN(C(=O)C(CSC)OC)C2)CC)=O)cc2c(s1)CCC2 C1(N(C(c2c(OC)csc2)=O)C)CCCCN(C(=O)Cc2cscn2)C1 CC(C)(C(=O)N1CCC(C(C)(O)CNC(C2CC2(Cl)Cl)=O)CC1)C(F)(F)F c1(C(=O)OC(C(=O)OC)c2cscn2)ccc(C(F)F)c(Cl)c1 CC1(C)CCOC1C(=O)NC(c1cccnc1)C(=O)NCc1cnsc1 N1(C(CC2(OC)CCCCC2)=O)CCC(NC(c2cc(C(N)=O)cs2)=O)C(O)C1 c1(C(N(C2CCN(C(C=C(C)C)=O)C2)CCO)=O)cn2c(n1)COCC2 C1(C(C)C(=O)N2CCC2CC2CCCC2)CCCN(C(c2ccco2)=O)C1 C12(C(=O)NC3CN(C(C=C(C)C4CC4)=O)C3)CCC(N=[N+]=[N-])C1C2 C1(NC(c2nc(C)sc2)=O)CC2CC1CN(C(=O)CC1CCCCC1(C)C)C2 C1(NC(CCC)=O)CC(O)(CNC(C2CC(C)(C(=O)OC)C2)=O)C1 c1(NC(=O)Cn2cc(Cl)cn2)nc2ccc(-c3cnn(CC4CCC4)c3)cc2s1 CCC(CC)(CC)C(=O)NC(C1CCOC1)CNC(C1CC(=O)NC(=O)N1)=O C#CCC(CC#C)C(=O)N1CC2(CCC(CNC(c3cc(CO)oc3C)=O)O2)C1 C1(N(C(=O)C2=CCSC2)C)CCCC2CN(C(c3c[nH]nc3C3CC3)=O)CC12 Cn1nnc2c(N3CCC(C(C)(C)NC(=O)Cn4cc(C5CC5)nn4)C3)ncnc12 N1(C(C2(CC)CCNC2=O)=O)CCN(C(c2cc(Cl)no2)=O)C(CC(F)F)C1 c1(C(=O)NC(C2(O)CN(C(C(C)OC3CCCC3)=O)C2)C)ccc(Cl)c(Cl)c1 C12(CNC(C(C)NC(N)=O)=O)CC1CN(C(=O)C=CCOC1CCOCC1)C2 Cc1ccc(CC(=O)NC(C)CC2CN(C(c3cc(=O)c(C)c[nH]3)=O)C2)cc1C CCN=c1[nH]c(C(=O)NC2CC3CC(NC(c4coc(C5CC5)n4)=O)C2C3)cs1 C(=O)(C(C)C(C)C)N(CC(C)C)CC(=O)N(C)CC1(NC(N)=O)CC1 C(=O)(CC(F)(F)C(C)C)N1CC(C(C)NC(c2c(C)cco2)=O)OCC1 c1(C(N(CC(C)NC(C=CCOC)=O)C)=O)ccccc1-c1nnc(C)o1 N1(C(C(COC)Cl)=O)CCC2CC(C1)CN(C(c1ccc(F)c3occc13)=O)C2 N1(C(C)C(=O)NC2CC(F)(CNC(c3csc(Cl)n3)=O)C2)CCC(O)CC1 c1(-c2ccc(OC)cc2)nc(N2CCC(C)C2CO)cc(N)n1 C1(CC)(NC(=O)CC2CCCC(=O)N2)CCN(C(c2cnn(C)c2OC)=O)CC1 c1(C(N2CCC(NC(C(CC=C)CC)=O)C(CO)C2)=O)cnc2c(c1)COCC2 N#Cc1ccc(C(=O)NC2CC(NC(=O)C(c3ccc(OCC#N)cc3)O)C2)o1 N1(C(C=NOC)=O)CCC(CC(C)NC(=O)CC2CCC3CC23)CC1 C(=O)(CC(C)CC(C)C)Nc1nc(Cc2cccc(OCCCCCCC)c2)sc1 N1(C(C2CC(C)(C)C2)=O)CCCC(F)(C(N2CC3CCC3(CO)C2)=O)C1 N1(C(C(N2CCC(C)C2)=O)=O)CCC(OC(=O)Cc2cccs2)CC1 C1(C(=O)NC2(COC)CC2)(NC(=O)C(c2ccccc2)F)CCN(C)C1 c1(C(N(CC(CN(C(c2c(C)nn(C(C)C)c2)=O)C)O)C)=O)cc(F)ccc1N C1(C(N(C2CCCN(C(c3ccc(C#N)o3)=O)C2)CC)=O)CCCCC1(F)F CCC(C)CC(C)C(=O)NCC(C)NC(c1ccc2c(c1)OCO2)=O Cc1onc(C(N2CCCC(NC(c3cc(F)cc(F)c3O)=O)C2)=O)c1[N+](=O)[O-] C1(F)(CNC(C(c2cncc(F)c2)C)=O)CCC(CNC(C2CC=CC2)=O)C1 C1(CNC(C(C)c2ccsc2)=O)CC(F)(F)CN1C(c1ccn(C)c(=O)c1)=O N1(C(COCCOCC#C)=O)CC(C(N2CC(C#N)(SC)C2)=O)CC(C)(C)C1 N1(CC(=O)NCCOCC#C)CCCCC1 C12(NCC(C(C)(O)C3CCOCC3)O)CC=CCN1CCC2 C(=O)(CC(C)(C)C(C)(F)F)NC(CCNC(C(COC)OC)=O)C C1(C(=O)N(C)CC2(NC(c3cnc(C(F)(F)F)s3)=O)CC2)(OC)CC(C)C1 C(=O)(C1=NNC(=O)C1)NC(CC(=O)NC(CC=C)C1CC1)CC1CC1 c1(OC)cc(C(N2CCC(NC(c3cccc(O)c3)=O)C(F)C2)=O)cc(O)c1O Cn1ncc(C(=O)NCCC2CCC(NC(=O)C=C3CC3)C2)c1CN1CCCC1 C(C(C)C(=O)N(C)CC1CCOC1)N(C(C(C)OCC(C)C)=O)C C1(CNC(C2CN(CC(F)(F)F)C2)=O)COCCN1C(C1CCOC1C1CC1)=O c1(OC)ccccc1S(=O)(=O)N1CCCC1CNC(c1nc(Br)cs1)=O c1(C(=O)NC(CC(=O)NC(C#C)(CO)CO)C2CC2)cccc(F)c1F c1(NCCN(C(=O)CCSC(F)(F)F)C2CCS2=O)ccn(C2CCOCC2)n1 CCC(C)C(O)C(=O)NCc1cc(C(N2CCC3C(C(N)=O)C23)=O)cs1 c1(CCC)cccc(C(=O)NCC(C2CC2)N(C(=O)C(O)C2CCC2)C)c1 c1(C2(C(=O)NCCC(C)(C)NC(=O)CO)CC2)ccc(Cl)nc1 Cc1ccnc(C)c1C(=O)NC1CC(C(F)F)(NC(C2CCC(C)O2)=O)C1 C1(NC(CCN(C(C(CCC)OC)=O)C2CC2)=O)CCN2CCCC2C1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(C2CCC(C)CC2)=O)cn1C C(=O)(C(C)O)NCCOCCOCCNC(C1(CCC)CC1)=O.C(C)(=O)N c1(C(N(CCN(C(C2CCCN(C)C2)=O)C)C)=O)ccc(N)cc1O C(c1ccccc1C)=CC(N1C(CN(C(CS(CC)=O)=O)C)CCC1)=O N1(C(C2(N(C)C(C3(n4cnnn4)CC3)=O)CC2)=O)CC2CCC2(C)C1 c1(-c2ccccc2)cncc(Br)c1.C12CCCN1C(=O)NC21COC1 c1(C(=O)NCC(CC=C)NC(=O)CC(C)n2cccn2)cccc(C)c1[N+](=O)[O-] N1(C(c2c(C)ccc(O)c2)=O)CC2OCC(NC(c3cc(Cl)cnc3C)=O)C2C1 C1(C(=O)NC2C(CCC)C2)(OC)CCN(C(C2CCCC2O)=O)CC1 C(=O)(C(C)(O)C(C)c1ccccc1)NCC(CC(C)C)NC(=O)CN(C)C(C)C C(C(C)=Cc1ccccc1)(C(=O)NC1CCCC1)N(CC)Cc1ccccc1 c1(C(=O)NCC2(CNC(C3C(C(=O)OC)C3)=O)CC2)c[nH]c2nc(F)ccc12 C1(CCC(=O)NC(COC)CNC(=O)CSC2CCOCC2)CCC(C)O1 C=CCC(C(=O)NCC1(OC)CN(C(C2CCCN2C2CC2)=O)C1)OC CN1CCc2cc(C(=O)NC3CN(C(=O)CC4CC5(CCC5)C4)C3)ccc21 C1(C(=O)NC(c2ncc[nH]2)C)(CNC(c2ccon2)=O)CCCCO1 c1(OC)cccc2c1CN(C(=O)C(=O)NCC)CCC2.C1(OC)CCCCCC1 c1(OCC(=O)NC2CC(CO)N(C(=O)CCC3CCCC3)C2)cccc(Cl)c1 c1(C(N2C(CNC(CCc3ccc(C)cc3C)=O)CC2)=O)ccc(Cl)c(C#N)n1 c1(C(=O)NC2CCCN(C(CCNC(=O)NC)=O)C2C)cnc2n[nH]c(C)c2c1 Cc1cn(C)nc1C(N1CC=CC1(C)C(=O)NC1CCC(F)(F)C1)=O N1(C(CCc2scc(C)c2)=O)C2CCC1CC(N(C(=O)Cc1nnc(O)s1)C)C2 C1(CCC(=O)NC(c2cnccn2)C)CCCN1C(c1csnc1Cl)=O c1(OCC(N)=O)ccc(C(N2CCC(CF)(NC(c3cscn3)=O)C2)=O)cc1 C(CCN(C)C(c1ccc(-n2ccnc2)nc1)=O)(C(C)C)NC(C(CC)C)=O CC(Cc1ccccc1)C(=O)NCCC1CC(Nc2ccncn2)C1 C=C(Cl)C(=O)NC1CC(N(C(C)=O)C(C2(c3nccs3)CC2)=O)C1 c1(C(=O)NCC2C(NC(CC3(C)CC3)=O)CCCC2)noc2c(F)cccc12 C1(NC(Cc2c(C)scc2)=O)CN(C(=O)C(C)Oc2ccccc2F)CC12CC2 c1(Nc2c(C(N)=O)c[nH]n2)ccc(S(=O)(=O)C(F)(F)F)cc1Br N1(C(C2CC(C)N2C(C2CC(=O)N(C)C2)=O)=O)CC=CC(CO)C1 Cn1ncc2nc(O)c(C(=O)NCC(CNC(c3cccc(O)c3)=O)CO)cc12 CCC(C)CCC(=O)N(C1CCN(C(=O)CC2CCCOCC2)CC1)CCO N1(C(=O)NCC(c2ccc(C#N)cc2)(C)OC)CC(C)CCCC1C C(=O)(C1OCCc2ccc(C)cc21)NCCCCCN(C(CC(=C=C)C)=O)C c1(CNC(C2CC3CC2C3)=O)nnc(O)n1C1CC1 CC1(C)CCOC(CNC(=O)CCC2CCN(C(=O)C(CO)NC(N)=O)C2)C1 c1(OC)cc(C(N2CCC(CO)(NC(c3cc(C4CCC4)no3)=O)C2)=O)ccn1 c1(C(N2CC(CCOC)N(C(=O)C(C)COC(C)=O)CC2)=O)cccc2sncc12 CC1=C(C(=O)N2CC(c3nc(C)no3)C2)SCCO1.C12CCN(CC1C)C2=O Cc1ccsc1C(c1nnnn1CCC1(C)CC1)NCc1ccnn1C(C)(C)C c1(C(N2C(CNC(CC3C(C)(C)C3)=O)CCCCC2)=O)cc2c(Cl)cncc2s1 C123CC(C1)(C(C)(C)O2)C3.C(=O)(CCCC(F)F)NCCOC1CCN(C(C)=O)C1 c1(C(N2CCC(CNC(c3[nH]cc(CC)c3)=O)C2(C)C)=O)cc(C)c(C)cc1C N1(C(c2cc(CSC)c(C)s2)=O)CCCC(O)(CCNC(c2ccco2)=O)C1 c1(NC(N2CCC(SCC)CC2)=O)cc(O)c2ccccc2c1 N1(C(=O)C(F)C(C)C)C2CCC1CC(C)C2.C1(OCC)CC2(C1)CC2CC=O c1(C(=O)NCC(CNC(c2ccc(CNC(C)=O)s2)=O)C)ccc2nonc2c1 C1(NC(=O)COCC2CCOC2)CCC2(CCN(C(=O)Cc3ccon3)CC2)C1 C1(C(N(C)CC2CCCO2)=O)COCCN(C(c2sccc2F)=O)C1 C1(C(=O)OCCCN(C(C)CCO)C)C2CC2CN1C(=O)Nc1ccccc1 C#CCN(OC)C(=O)CC1(CNC(c2cc(=O)cc[nH]2)=O)CC1 C1(O)(CNC(CC2C(C(=O)OCC)CC2)=O)CCC(C)(C)C1 CC1(C)CCC(C(=O)NCC(CNC(=O)CNC(N2CCCC2)=O)CO)OC1 C1(C(=O)NCC(C2CCN(C(C=CC)=O)CC2)O)(OC)CCC(C)(C)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)N1CC(C)N(C(C2CC2C(F)F)=O)CC1 C#Cc1ccc(CNC(=O)CC2C3CN(C(=O)C(C)NC(=O)CC)CC23)cc1 C(=O)(C1CSc2ccccc21)NC(C1(O)CCN(C(=O)Cn2ccsc2=N)C1)C N1(C(CC2CC(CC)C2)=O)CC(=O)NCC1C(=O)NC(CC1CCC1)CO N1(C(CCOCCC)=O)CCCC(CCCCNC(C2(O)CCC2)=O)C1 N1(C(c2ccn(CCC)n2)C(=O)NC(C)C)CC=C(c2ccccn2)CC1 C1(CN(C(c2c(C)nsc2)=O)C)CCN(C(=O)C(C)(O)Cc2ccccc2)CC1 C1(C(N(Cc2cnc(C3CC3)nc2)CCC=C)=O)Cc2cc(C)c(C)cc2O1 C(=O)(C(C#N)C(=O)CCc1cccs1)N(CCOC)Cc1ccccc1 C(=O)(C1CCCc2scnc21)NC(CCN(C(c1ccc(C)o1)=O)C)C CC(CNC(=O)CC1CC1(Cl)Cl)CN(C(=O)CNC(c1ccsc1)=O)C CN=c1nc(N2CCC(N(C)C(=O)NC)C2)[nH]c(=NC2CCC(F)CC2)[nH]1 CCC(C)C(O)CC(=O)N1CCCC(CCC(=O)NCCC2CCC2)C1 Cc1cnn(C)c1CC(=O)NCC1CC1[N+](=O)[O-] c1(C(=O)NCC(CNC(c2ccc(C)o2)=O)C)cc(F)c(C(F)(F)F)c(F)c1 C1(O)(C(=O)NCC(CNC(C(c2n(C)cnn2)(C)C)=O)CO)CCCCCC1 c1(N(C2CN(CC(F)F)C2)C(Cc2cn(CC)nc2)=O)ccc(C)c(C)c1 C1(NC(C(C)NC(N)=O)=O)CC2CCC1CN(C(c1cccs1)=O)C2 C(C(F)C(=O)N(C1(O)CN(C(=O)COc2cc(C)on2)C1)C)N(CC)CC CC(C)(CCC(=O)NC1COCC1CNC(=O)CCc1cn[nH]c1)[N+](=O)[O-] C1(NC(c2cn(CC)nc2)=O)C2CCCN(C(=O)C(C)n3ccnn3)C2C1(C)C C12(NC(c3c(OC)c(C)cs3)=O)CCC(CC1NC(=O)C(C)S(N)(=O)=O)C2 C1(NC(C2(NC(COCC(=O)NC)=O)CC2)=O)CCC2(CC1)CC(OC)C2 C1(C2(C)CC2)(C(=O)NC2(C(=O)O)CC(C)C2)CC1 CCC(CC)C(C(=O)NCCCCC(C)NC(C1CC(OC)C1)=O)OC Cc1cc(=O)ccn1CC(=O)NCC1CCC(NC(C2(C#N)CCSCC2)=O)C1 N1(C(c2cnc(CC(C)(C)C)o2)=O)C2CCC1CN(C(=O)CC1=CCCC1)C2 C1(C(F)(F)F)CC(N=c2nc(N3CCCOCC3)c3c([nH]2)CCCC3)C1 C1(C(N2C(CNC(c3cccc4cnnn34)=O)C=CC2)=O)CCCC(F)(F)CC1 c1(-c2n(-c3ccc(OC)c(Cl)c3)nc(-c3cncnc3)n2)cc2ccncc2[nH]1 Cc1cc(C)nc(CCN(C2CCN(C(=O)OC(C)(C)C)CC2)C2CCO2)n1 C1(NC(C2CN(C(C)=O)C2)=O)CC(NC(=O)C(C)(C)n2cnc(C)c2)C12CCC2 N1(C(c2nc(C)[nH]n2)=O)CCCC12CCN(C(C1(C)CC1(Cl)Cl)=O)C2 C1(C(C(=O)N(CC(=O)N(CC)CC)C)C)CCCOC1.C1(=O)CN1.C(C)(=O)N c1(NCC)cccc(C(=O)NC2CCCC2NC(c2cnc(OC3CC3)s2)=O)c1 c1(SCc2n(CCC)ncn2)cccnc1N1CCC(C(N)=O)C1.C(C(F)(F)F)N N1(C(=O)CC2CC(OC3CC3)C2)CCC2CCN(C(=O)CC3CCCCO3)CC12 C12(NC(CN(CC)CC)=O)CC1CN(C(c1nocc1Cl)=O)C2 C(=O)(CC1COc2cc(OC)ccc21)NCCCN(C(=O)Cn1cnnn1)CC c1(C(=O)NC(C(=O)NCCOC)c2cccs2)cn(CC2CC2)nn1.C1(=O)CN1 C(=O)(CCCC(=O)N1CC(CNC(=O)CNC(=O)OC(C)(C)C)CC1(C)C)NC c1(C(=O)NCC2(O)CCN(C(C3(C)CC4CCC3O4)=O)C2)cccn2nccc12 c1(C(N(CCNC(c2cc(CCO)on2)=O)CC)=O)cc(Cl)c2n[nH]cc2c1 c1(C(N2CCC(CNC(c3cc(C#N)oc3)=O)C2)=O)cc2scnc2[nH]1 c1(N2CCC(F)(CN(C)C)C2)nccc(=NCC2CC2)[nH]1 C12(C(=O)NC(c3ccccc3)CNC(c3cc(Br)co3)=O)CCCC1OCC2 C(C)(C)(CC(C)CO)NC(C1(CNC(=O)C(C)N(CC)CC)CC(=C)C1)=O N1(C(CCC(=O)NCC)=O)CCN(C(=O)C(C)C2CCC2)CC1c1ccnn1C C(=O)(CCCCCN=[N+]=[N-])N1CCC(C)(NC(C2OCC(C)C2)=O)CC1 c1(CC)ncc(C(=O)NCC(C)CNC(c2ccc(C)c(F)c2)=O)c(O)n1 C(C1CN(C(c2cccc[n+]2[O-])=O)CC1C(=O)N(C1(C)CCCC1C)CC)=CC N1(C(CC=C)=O)CCC(NC(C2CCCN2CCC)=O)C1(C)C c1(OC)cc(C(=O)NCC(=O)NCC=CCNC(C2CC2C)=O)[nH]n1 c1(C(N2CC(O)CC(NC(CC=CCC)=O)C2)=O)cc2cc(Cl)ncc2[nH]1 C(c1ccccc1[N+](=O)[O-])=CC(N1CC(NC(C(CC=C)C)=O)C(C)(C)C1)=O S(=O)(=O)(c1ccc(N2CCCC(OCC(F)(F)F)C2)cc1Br)N(CC(C)SC)C N1(C(COCC(C)C)=O)CCN(C(C2COC(=O)C2)=O)CC1c1ccccc1Cl c1(NCCCC(N)=O)cc(NC2COCCOC2)ncn1 C1(C(=O)NCCN(C(=O)C(C)SC(F)(F)F)CCC)CC2(CCCC2)C1 CN1C(=O)N(C2CCN(CC(c3cccnc3)O)CC2)C(=O)C1c1cccn1C C1(CC(=O)NCCC2CCN(C(C3CC(C)(F)C3)=O)CC2)CCC2(CCC2)CO1 c12ccc(Br)cc1C(=O)N2.C(=O)(C(c1cn[nH]c1)N(C)C)NCCOCC N1(C(CSCCNC(c2ncc(C(=O)OC)nc2)=O)=O)CCCC(O)CC1 N1(C(COCC=C)=O)CCC(NC(=O)CCC(F)F)C(C(F)(F)F)C1 N1(C(C(CN(C(CC(CC)C(C)C)=O)C)C)=O)CCc2ccc(F)cc21 C1(C(=O)NC2CC(NC(CC(=O)NCCNC(C)=O)=O)C2)CCC(C)(C)C1 c1(OC(C)C)ncccc1C(=O)NCC(C)N(C(=O)CC1C=NN(C)C1=O)C C12(C(N3CC(CC(=O)OC)OCC3)=O)CC=CC(C1)OC2.C1(C(=O)N)(CO)COC1 C1(F)(CNC(c2cnn3ccsc23)=O)CCCN(C(=O)C=CCF)C1 N1(C(CSC)=O)CCN(C(=O)C(N2CCOCC2)C)CC12CC2.CC(C)CO N1(C(Cc2scc(C)n2)=O)CC(CNC(=O)C(C)SC(F)(F)F)CC(C)(C)C1 C(=O)(C(C)C(O)C(C)C)NC(C(C)OC)C(=O)N(C(C)C(N)=O)C c1(OCC(=O)NCC2CC(NC(C=C(C)C3CC3)=O)CC2O)c(Cl)cccc1Cl C12(CNC(COC)=O)CCC1CCN2C(c1cc(=O)n(C)o1)=O C1(C(=O)OCc2ccnc(Br)c2)CN(C(=O)NC(C)(C)C)CCC1CO C(=O)(C1Cc2ccccc21)N1C(C)(C)C(CNC(=O)CSC2CC2)CC1 C1(NC(C(=O)N(C)C)=O)CC2(CCN(c3ncns3)CC2)CO1 Cc1c(C(N2CC(NC(c3cn(C)nn3)=O)CC(C)C2)=O)sc2[nH]cnc(=O)c12 c1(NC(C2CCCN(Cc3ccc(Cl)nc3)C2)=O)cccnc1OC(F)F c1(C(=O)NCC23C(CN(C(CC(C)(C)OC)=O)C2)C3)ccnc(C)c1Cl c1(CC(N2C(CCOC(C)(C)C)CCC2)C(=O)NC(C)(C)CC)ccc(F)cc1 CCCC(C(=O)NCC1(C)CCN(C(c2n[nH]c(=N)s2)=O)CC1)S(N)(=O)=O c1(C(N2CC(CC)C(Nc3ncncc3C)CC2)=O)cc(F)c(F)c(F)c1 Cc1ncc2ccc(C(=O)NCC(C)NC(=O)CCCc3cnn[nH]3)cn12 c1(C(=O)NCC(c2cccc(C)n2)(C)C)cncc2cccnc12 C(=O)(C1=NN(C)C(=O)CC1)NCC1(O)CC(NC(CCC(C=C)(C)C)=O)C1 CCCC(C#N)C(=O)N1CCN(C(=O)C=CBr)C(CC2CC2)C1 c1(C(N2C(CCNC(CC=CC=C)=O)COCC2)=O)nccc2n[nH]cc12 C(=O)(C(CC(F)F)NC(=O)C=CCN1CCCC1)NC1(CC(=O)OC)CCC1 c1(CN(C(c2ccc(F)cn2)C(=O)NCCC2CC2)C)ccc(OC2CC2)cc1 C(=O)(C(O)CCn1cncn1)NCC(C(C)C)NC(=O)C(C)(C)F c1(OC)ccc(NC(N2CCSC(C(F)(F)F)C2)=O)c(Br)c1 N1(CCC(C)(C)NC2C(CC)COC2)CCC(C)CC1.C12CCCC1NC(=O)O2 C(CCC(=O)N1CC(O)(CNC(=O)CN(S(C)(=O)=O)C)C1)N(C(C)C)C c1(N(CC)CC)cncc(C(N2CCOC(CNNS(=O)(=O)C3CC3)C2)=O)c1 c1(C(N(C)CC2(O)CCCN(C(COCCOC)=O)C2)=O)cc(N)c(C)cc1C N1(C(C2CCC(NCc3cccc(CO)c3)C2)=O)CCN2CC(O)CC2C1 C1(NC(C2CCN(CC)C2)=O)CN(C(=O)Cc2cncc(C)c2)CC2(CCC2)C1 C(CC1CCCC1)(C(=O)NCCCN1CCC1)NC(=O)CC1CCOC1 c1(C(N2C(C)CC(NC(=O)C#CC3CC3)CC2)=O)c(F)ccc(F)c1N N1(CC)CCN(CC(N2CC(CNC(=O)Cc3ncc(C)s3)C(C)C2)=O)CC1 CC1(C)CCC(CC(=O)NCC2CCCN2C(=O)CCOC2CCOCC2)OC1 N1(C(c2c(C(C)(C)C)ncs2)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC1CO C1(CCC)(NC(=O)CC(F)(F)F)CCN(C(=O)C(O)C(C)SC)CC1 C1(CNC(C(C)C2CCC2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1O c1(CN2C(C(=O)Nc3c(C(C)(C)O)cccc3)CC(O)C2)c(Cl)cnc(Cl)c1Cl C(=O)(C1CCc2c[nH]nc21)NC1C(NC(CCc2ccc(=N)[nH]c2)=O)CC1 c1(CCc2nn[nH]n2)cnccc1C(N1CCC(CCSC)C1)=O c1(C(=O)NC(CC(C)NC(C(CC)CO)=O)C)ccc(OC)cc1Cl c1(C2OCCN(CC(=O)Nc3nnc(C(C)(C)C)s3)C2)cccc(Cl)c1Cl c1(C(N2CCC(NC(C3(C)CC(C)(C)C3)=O)C2)=O)ccc2occc2n1 N1(C(CCCn2ncc(C)c2)=O)CCN(C(=O)C(Cl)=CCl)C2CC12 c1(C(N2CCCCC(NC(C=C(C)Cl)=O)C2)=O)ccc(=O)n2c1CCCCC2 N1(C(c2c(NCC)cccn2)=O)CC2(CCCC2NC(=O)C(C)CC)C1 C1(N(C)C(c2cnn(C)c2)=O)CCN(C(=O)C(c2ccccc2)F)CC1 c1(CNC(C=C(CC)C)=O)ccc2c(c1)CCCC2NC(C1COCCN1C)=O c1(C(N2C(C3(O)CCN(C(c4cc[nH]c4)=O)CC3)CCC2)=O)ccc(F)c(Cl)c1 c1(OC)coc(C(=O)NCC2CCCC(NC(c3cccc(F)c3)=O)C2)cc1=O c1(C(N(C2CCN(C(C(C(C)C)(C)C)=O)C2)CCO)=O)cc2cccc(Cl)c2[nH]1 N1(CC(=O)N(CC(C)C)CC(N2CC(C(=O)NC3CC3)C2)=O)C(=O)CCC1=O CCCC(O)(CCC)CC(=O)NC1CCC(NC(c2cn(C)c(C)cc2=O)=O)C1 C1(CC(=O)N(C(CN(C(CNC(CC)=O)=O)C)C)C)CCC(C)(C)CO1 c1(OC)ccc(NCc2ccc(O)c(C(=O)OC)c2)c2ccccc12 c1(C(N2C(C(N(C)Cc3ncnn3CCF)=O)CCC2)=O)ccc(C#N)cc1 c1(C(=O)NC2CN(C(C(F)=CCC)=O)CC2C)ccc(-n2nccc2C)c(F)c1 CC(CC(C)(F)F)C(=O)N1CCC(NC(c2c(N)cc(Cl)cc2Cl)=O)C1 N1(NCc2cc(OC)c(OC)cc2)CC2CN(C(c3sccc3C)=O)CC2C1 C12CCOCC1NC(=O)N2.C1(SC(C)(C)C)CC(C)N(CCC(C)C)C1 C1(CNC(C2(C)CN(C)C(=O)C2)=O)CC12CCN(C(C1CC(F)(F)C1)=O)CC2 c1(CCC(=O)NC2CCN(CCCC3CCOC3)C2)ccc(O)nn1 c1(C2C(C(N3CC(OC)C(NC(c4nnn(C)n4)=O)C3)=O)C2)ccc(Cl)c(Cl)c1 CCCC(C(=O)OC)C(=O)NCC1CCC(NC(C2CCOC(C)(C)C2)=O)C1 N1(C(C(C)OC2CCOC2)=O)CCN(C(c2cc(CO)on2)=O)CC1CC(F)F C(=O)(C1=CCCOCC1)N1C(C)C(C(=O)NC23CC2COC3(C)C)CCC1 N1(C(C(C)OCOC)=O)CCC(CC(N2CC(OC(F)F)C2)=O)C1 C1(C(=O)NCCCCC2CN(C(COC(CC)C)=O)C2)CC(C)(C)CN1C C(=O)(C(CC1COCCO1)C(F)(F)F)N1CC(NC(C(=O)NCC)=O)C(C)C1 c1(CC(N2CCN(C(COC)=O)C3C2CC3)=O)ccc2c(c1)CCCO2 C1(c2n(-c3cccc(OC)c3)nnn2)(N(C2CCCCCC2)C)CCCSCC1 CC(C)(C)CCC(=O)NCC(=O)NCC1(F)CN(C(C2CCCO2)=O)C1 N1(C(C=CC=CC)=O)CCC(N(C)C(c2cc(C(F)(F)F)c[nH]2)=O)C(C)C1 Fc1cc(CNC2(c3nnnn3C3CCOC3)CCOC2)c(F)c(F)n1 N1(C(C(CC=C)NC(C)=O)=O)CCC2(C1)CN(C(C1CN(S(C)(=O)=O)C1)=O)C2 c1(C(=O)NCC2CC(NC(CCCc3onc(C)n3)=O)C2)[nH]c(C)c(C)c1C C1(C(=O)NC2CCC(N(C(C(C)COC(F)(F)F)=O)C)CC2)CCC(=O)N(C)C1 Cc1ncccc1-c1cn(CC2C(CNC(C3CCCC3CF)=O)C2(F)F)nn1 N1(C(C2C(CC)C2)=O)CCOC(C)(CNC(c2ccc(-c3ccccc3)n2C)=O)C1 c1(N(C(c2coc(C)n2)C(=O)NCSc2cnn(C)c2)CC)cccc(OC)c1 N1(C(c2c(C)nn[nH]2)=O)CCCC(C(C)NC(=O)CCc2ccon2)C1 c1(C2CC(Cl)C2)ccccc1-c1ccc(C2CCCCO2)cc1 C1(OCc2ccc(OC)cc2)CC2CCCN2N1CC1CC2CCC(C1)N2C C(=O)(CC(C)(O)C(F)(F)F)NC1C(CCCCNC(CN(C)CCO)=O)C1 c1(NC(C)=O)ccccc1NC(=O)C(=O)NC1CC(SC2CCOC2)C1 c1(OCCC)cccnc1C(=O)NC(C)CCNC(c1cnc(OCC)s1)=O C(=O)(C1CCCc2c[nH]nc21)N(CCCCCCNC(C(CCC(C)C)O)=O)C c1(NCC2C(C)CN(C(=O)CCn3cnnn3)CC2)ccc([N+](=O)[O-])cc1CO N1(C(C(C=CC)O)=O)CCN(C(c2cc(O)cnc2N)=O)C(C)C1 C(=O)(C1=Cc2ccccc2OC=C1)NCC(CN(C(Cc1c(C)ccs1)=O)C)O c1(CC(=O)NCC(CC)(C)NC(C2CCCCC2O)=O)ccc(S(C)(=O)=O)cc1 N1(C(C=CCC)=O)CCCC(C2CCN(C(=O)C(O)CC3CC3)CC2)C1 C1(NC(C(C(CC)C)O)=O)CC2CC1CN(C(c1ccc[nH]1)=O)C2 C1(C(=O)NC(Cn2ncc(C)c2)C)CC(=O)N(c2cccc(C(F)(F)F)c2)C1 CN1C(=O)CSC1=CC(=O)NC1CC2(C1)CC2NC(C1CCCCC12CCC2)=O C(CCCCCC(=O)NC(C)(C)CCNC(C1CC12CC(F)(F)C2)=O)SC c1(SC)ccc(CC(C(=O)OC)NC(c2scnc2C)C)cc1 C(CS(=O)(=O)CC(=O)NCC=CC(=O)NC(C)Cc1cccs1)OC C=CC(C)(C)C(=O)NC(CN(C(=O)CC(C)CF)CC)CC.C(C)(=O)O c1(SCC(N2CCC(C)(CNC(C3CCC(=O)N3)=O)C2)=O)ncnc2[nH]cnc12 N1(c2nc(C)c(C#N)cc2)CC2CCCN(C(=O)C(C)CF)C2C1 CCCCCC(=O)N1CCC1CNC(C1CC2CC2C1)=O.N12CCC(CC1)C2=O c1(C(=O)NC23CCN(C(CC(C)C(C)(C)C)=O)CC2C3)nc2ccccn2c1F C(=O)(N=c1cc[nH]c2cccnc12)c1cc(N2CCN(CC)CC2)ncc1 c1(NC2CC23CCC(NC(=O)C=CBr)CC3)ccc([N+](=O)[O-])cc1.CC1C(=O)N1 N(C(=NCCOC1CCSCC1)Nc1ccc(Cl)cc1)C1CCC(=O)NC1 Cc1cccnc1C(N1CC2CC2(CNC(=O)C(C)OC2CCCC2)C1)=O C1(NC(=O)CC2CC2)C2CCC1CN(C(=O)C1=NOC(C3(O)COC3)C1)C2 c1(NC(=O)NC(CC)C(N2CCC(C)(CCO)C2)=O)ccc(O)c(F)c1 C1(C(=O)NC2(CCCNC(CNC(COCC)=O)=O)CC2)CC(C)(C)C1C(C)C N1(C(C2(OCC)CCCC2)=O)CCCC(C2CCN(C(=O)CC3CC=CC3)C2)C1 C1(CNC(C2OCCN(CC)C2)=O)CC2(CC2)CN1C(C1OCC1(C)C)=O N1(C(c2cn(CC)nc2C)=O)CCCN(C(c2cccc(OC)n2)=O)C(CO)C1 N1(C(C)=O)CCCC(C(N2CCC(O)(CNC(=O)CSC3CC3)C2)=O)C1 C1(C(=O)NCCN(C(C2OCCC2C(C)C)=O)CC)CCOC2(CCC2)C1 C(=O)(CCCC(c1nnnn1C)NC1CCCCC1c1cccc(C)c1)OCC C=C1CCN(C(=O)CCCCN(C)C)C(C(=O)Nc2ccc(N(C)C)cc2C)C1 C1(NC(C(CCOC)NC(=O)CN2CCC(F)CC2)=O)C=CC(C)(C)CC1 C12=CC=C(C=C1)C2.n1(CCNC(CNS(C)(=O)=O)=O)cc(C2(O)CCOC2)nn1 C1(CNC(C2C(C)C2)=O)CCCN(C(=O)CC2(CO)CC2)C1 C1(C(C)C)CCN(C(=O)C(C2CC2)N(C(=O)CC2(O)CCC2)C)C1 C(CNC(C1CNC(=O)C1)=O)(CC(F)(F)F)NC(CS(=O)(=O)NC(C)(C)C)=O C12C3CN(CC13)C(=O)C13CC(CN1C2)C3.C12(CC(=O)N(C)C)CCCC1C2 c1(CC(N2CCC(N(CC#C)C(c3ccc(F)o3)=O)C2)=O)ccc(F)cn1 C1(NC(C2NC(=O)CC(C)C2)=O)CC2CC(C1)N(C(=O)CN1CCCNC1=O)C2 N1(C(CCCC(C)=O)=O)CCC(C2CCN(C(C3CCS(=O)(=O)C3)=O)CC2)C1 S(=O)(=O)(c1cnc(NCC2(C)CCCC2)c(Cl)c1)N(CC(CCC)O)C N1(C(c2n[nH]c(C)c2Cl)=O)CCN(C(C2CN(C)CC(C)O2)=O)CC(O)C1 CC(C)CCC(O)C(=O)N1C2CCC1C(C(=O)NCC1CC(C)(C)CCO1)C2 CN1CCC(C(=O)NCCc2ccnc(-c3cccc(C(N)=O)c3)c2)CC1 c1(OC)ccc(Br)c(F)c1CN(C)C(C)=O.C12CC1C(=O)N2 CC(CN(C)C)CCC(=O)NCC1(O)CCCN(C(=O)COCCCN(C)C)C1 Cc1ccc(C(N2CC(OCCNC(=O)Cc3cncnc3)C2)=O)cc1[N+](=O)[O-] C1(CCC)(C(=O)NCCC(=O)NCCOCc2cc(C(C)C)on2)CC(=O)C1 c1(OC)c(F)ccc(C(=O)NC2C3CCC2CN(C(C2(N)CCC2)=O)C3)c1F CCCCCCC(C)CC(=O)N(CCCNC(=O)CCC1CCOCC1)C(C)C CCCC(O)CC(=O)N1CCN(C(=O)C(C)=C2CCCC2)CC1c1nccn1C C12(C(N3CCC(C(C)(C)NC(c4cc(O)ncn4)=O)C3)=O)CC3CC1C2C3O c1(CN=C(NC(COC)C)NC2CC2(C)C2(C)CC2)ccc(C#N)c(F)c1 C1(NC(C2CCC(C)C2)=O)CC2CCCC(C1)N2C(C1CC(C)C1)=O C1(n2cc(-c3c(C(=O)OC)nccc3)nn2)CCC(C)(C)N(C(=O)C(F)OC)C1 C1(N=[N+]=[N-])(C(=O)NCCCc2nc(C)[nH]n2)CCN(C(=O)C#CC2CC2)C1 N1(C(C(COC)(C)COC)=O)CC(CO)C2(C1)CN(C(c1csnn1)=O)C2 C[S+](C)CCC(O)C(=O)N1CCC(C)(CNC(=O)C(C)(C)NC(=O)C(F)(F)F)C1 c1(NCc2c(OC(C)C)cccc2)[nH]c(=NCCS(N)(=O)=O)nc2c1ncn2C CCC(C)CC(=O)N1CCCCC1N(C)C(c1cc(SC)ccn1)=O N1(C(CC(C)(C)C#N)=O)CCC2(CC1)CN(C(=O)Cc1ccon1)C1COCC21 Cc1cc(C(=O)NCCC2CC(NC(=O)COC3CCC3)C2)c2ncccc2c1 c1(C(=O)OC)c[nH]c(C)cc1=NCC(CNC(=O)CCCCCF)C(F)(F)F C(=O)(CC1OCCc2ccccc21)N1CCC(F)(CNC(C2CCCO2)=O)CC1 N1(C(CC(CC)C)=O)CCC2CN(C(=O)CCCCCOC)CC2CC1 C1(NC(c2cc(Br)n[nH]2)=O)CC1C1CCN(C(=O)COc2ccon2)CC1 C(=O)(C(C)CC(F)(F)F)NC(CN(C(c1cncnc1C)=O)CC)C c1(C(N(CC)Cc2cn(C3CCCC3O)nn2)=O)ccnc2[nH]ncc12 C=CCC(C(=O)NC1COCC1CNC(=O)Cn1cccc1)c1ccccc1 CC1(C)CC2C(CN1C(=O)C(=O)Nc1c(I)ccnc1Cl)C2(F)F Cc1cccc(C(CNC(=O)C(c2ccnn2C)O)NC(c2csc(C)c2)=O)c1 N1(C(c2scc(C)c2C)C(=O)Nc2ccccc2)C2CCCC1COC2 C1(N(C)C)CCN(C(=O)CCN(C(=O)CN(c2ccccc2)C)CC2CC2)C1 N(C(=NCC1CCC(C(N)=O)CC1)NCC(F)C(F)(F)F)CC(C)(C)C N1(C(C(CC2CCCC2)NC(=O)CC2CCCO2)=O)CCC(CCCC2CC2)CC1 C1(C(=O)NC2C(=O)NOC2)CN(Cc2cc(F)c(Br)c(F)c2)CC(F)(F)C1 N1(C(c2c(C)cc(CO)o2)=O)CCN(C(=O)CN(C)C2CC2)C2CS(=O)(=O)CC12 C(CCC(C)C(=O)N1CCC(C(C(C)C)NC(C2(C(N)=O)CC2)=O)CC1)OC C(=O)(CCCC(=O)NC1CCC(C(=O)N(C)Cc2cn(C)nc2C)CC1)OC C=C(C)c1ccccc1NC(=O)CCC1(C)CN(C(=O)CCN(C)CC)C1 C(C1=Cc2ncccc2C1)N1CC(=O)N(c2nc(Cl)c(Cl)nc2CO)C1=O c1(C(=O)NCCN(C)C(C2COC(=O)O2)=O)cc(=O)c2ccccc2o1 c1(NC)nnc(-c2cccc(N3CCCC3)n2)n1Cc1cccc(CO)c1 C1(C(C)NC(C(F)=C(C)C)=O)CCCN(C(c2ccc(C(C)=O)cc2)=O)C1 C1(NC(CC(=O)NCC#C)=O)(CNC(=O)Cc2cnc(C)[nH]2)CCOCC1 C(c1ccc(C)nc1)=CC(=O)NCCN(CCC)C(C1CCCCN1CCC)=O C1(Cc2c(OC)cccc2)CCN(c2cc(O)cc(F)n2)CC1C N1(C(C(C)n2cccn2)=O)CC2(C1)CN(C(=O)CN(C)C(=O)C1CC1)CC2CO N1(C(CCCc2ccc(CC)cc2)=O)CCN(C(=O)CCS(C)=O)C(C)C1 c1(C(C2CC2)NC(=O)NC2C(F)(C(=O)OC)C2)ccc2ncn(C)c2c1 CN1CCOCC1C(=O)NC1C=CCN(C(=O)CCCCc2ccccc2)C1 C1(CCNC(=O)Cc2ccsc2)CC(F)(F)CN1C(c1nnc(O)nc1O)=O C1(NC(C(C)C(C)O)=O)CCCC12CCN(C(=O)CCn1cncn1)CC2 c1(C(N(CC(C)N(C(=O)CC2CC2(Cl)Cl)C)C)=O)cc(Cl)ccn1 C1(CNC(C=C(C)C(C)C)=O)CCC2(CN(C(C3CC3C3CC3C)=O)C2)O1 c1(C(N(CC(CN(C(Cc2cc(C)no2)=O)C)O)C)=O)coc(S(C)(=O)=O)c1 C(C(C)(C)CC(C)(C)C)NC(c1cc(CNC(C(C(C)C)F)=O)[nH]n1)=O c1(CC(=O)NC(C(CO)NC(c2nc(CCC)oc2)=O)C)cc(Cl)n(C)n1 CC(C)C(CNC(C1(NC(c2ccc(F)c(F)c2)=O)CC1C)=O)C(C)C c1(CNC(C2CC(CF)C2)=O)cccc(NC(=O)CC2CC3CC3C2)c1 C1(CC)CC(C(=O)N(CCCNC(=O)C=C2CCCCC2)CC2CCCC2)CCO1 c1(C(=O)NCCN(C(=O)C(C)C(F)(F)F)CC(C)O)coc2c1C(=O)NCCC2 C(CC(=O)N1CCCC(CCF)C1)(C(F)F)NC(c1cn(C)nc1)=O C#CCC(CC(F)F)C(=O)N1CCC2CCC(C1)N2C(C1(CC)CCNC1=O)=O S(=O)(=O)(c1ncccc1Br)NC1CC(OCC)C12CCCCC2 N1(C(C(C)C(=O)NOCCCN(C)C)=O)CC=CC1CN(C)C C(=O)(C(O)CCC(C)(C)CC)N(CCC(C)NC(C(C=C)(C)C)=O)C O=C(C#CC1CCCO1)NCC1CCCN(C(=O)CC2CC2)C1 C1(C(C)C)CN(C(c2ccc(C#N)c(O)c2)=O)CCCN1C(=O)COCC(C)(C)C C1(C(=O)NCc2ccc(CO)o2)(COC)CN(C(=O)CC2CC2(C)C)C1 C1(NC(c2ncon2)=O)CCC2(CC1)CN(c1ncc(-c3ccccc3)cn1)C2 c1(C(N2CC(F)(CC(C)C)C2)=O)ccc(CNC(c2cc(CO)ccn2)=O)cn1 c1(CC(C)CN2CCOC(c3nnnn3CCCF)C2)ccc(O)cc1 c1(CC(=O)NC(C2CCC2C)=O)c(C)cccc1Br.C1(CC)CN(C2COC2)C1 C1(CC(N2CC(CC)N(C(c3csc(C)c3C)=O)CC2)=O)NC(=O)CN(C)C1=O c1(C(N2CCN(C(C3(CC=C)CC3)=O)CC2)=O)ccc2c(n1)CCC2 C1(C)(CC)CC(NC(c2cc(OC)ccc2F)=O)CN1C(=O)CCOC N1(C(C2N(CCC)CCC2)=O)CCC(NC(C2CC2C(C)C)=O)CC1 C1(C)(C(C)C)CN(C(=O)COc2cccc(CF)c2)CCO1 c1(C(N2C3CN(C(C(C(C)O)(F)F)=O)CC2CC3)=O)cnc2n1CCC(C)C2 c1(-c2cn(CCC)nc2)ccc(C(=O)NC(C)C)c2[nH]ccc12 S(=O)(=O)(c1cccc(C(C)(C)C)c1)C(=O)OC(C(C)C)C(=O)NCc1cnnn1C Cc1nc(N(C2CC3CCC(C2)N3)Cc2ccc(OC(F)F)c(F)c2)cc(O)n1 N1(C(c2c(N(C)C)nccc2)=O)CC2=C(C1)CN(C(C13COC(CF)(C1)C3)=O)C2 Cc1cccc(CC(=O)NCC2C=CCN2C(=O)CCOC(C)CC(C)C)c1Cl C1(C(=O)NC2C3CCC2CC3)CC2CCC(C1)N2 N1(C(CCN(CCC)C)=O)CCCN(CCNC(=O)C(=Cc2cnc[nH]2)C)CC1 C1(NC(C(CC=CC)NC(=O)CC2CCCN2CCC)=O)CNC(=O)C12CC2 C1(NC(c2cccc(OC(C)C)c2)=O)CN(C(c2ccc[nH]2)=O)C2CCCCC12 CC1(C(=O)NCCNC(C23CC(C2)C(C(F)(F)F)O3)=O)CCC(F)(F)C1 CC1=CC(C)CN(C(=O)CC2CN(C(C3CCN(C)C3)=O)CC2C)C1 C1(CNC(C(COC)OC)=O)COCCN(C(=O)Cc2cc[nH]n2)C1 Cn1nc2c(c1C(=O)NCCn1nccn1)CN(C(c1ccc(F)c(F)c1)=O)CC2 N1(C(C(CC=C)OC)=O)CC2(CC(CNC(c3ccc(Cl)c(C)c3)=O)C2)C1 C1(O)(CNC(C2(CC=C)CCC2)=O)CCCN(C(=O)CC(C)n2ccc(C)n2)C1 CCCCC(=O)C(=O)NCCCCC(=O)NCc1cc(F)ccc1F C(=O)(CC(C)(C)N(C(=O)CCOCC1CCCO1)C)NCC(C)OCC C(=O)(CC(C)C(C)(C)C)NCC1(OC)CN(C(C23CCC(CC2F)C3)=O)C1 c1(C(=O)NCC2(NC(C3C(C=C)CC3)=O)CC2)cc(Cl)c(O)c(Cl)c1 C(CCCC(=O)N(C)CC1(N(C)C)CC1)N(C(=O)C(C)(C)n1ccnn1)C c1(C(C(=O)OCC)O)cccc(NC(C2(NC(=O)C(O)CCSC)CCC2)=O)c1 Cc1c(Cl)ccc(C(=O)NCC2C(C)CCCN2C(c2nncs2)=O)c1N c1(OC)ccc(CC(=O)NC2CCOC(CNC(c3csnn3)=O)C2)c(OC)c1 Cc1cc(=NC2CCCS(=O)(=O)CC2)[nH]c(=NCC2CCCC(C)CC2)[nH]1 c1(C(=O)NC(C)CC(C)NC(c2ccc(O)c(O)c2)=O)ncn2ccccc12 Clc1nc2ccccc2cc1-c1nc(C2CCCCC2)nn1-c1ccncc1 N1(CCNC(C(CCN)c2c[nH]nc2CO)=O)CC2COCC2(CO)C1 c1(C(=O)NC2CC(N(C(C3CC(CC)C3)=O)C)C2)ccnc2[nH]c(C)nc12 c1(OC(C)C)ccc(CNCc2ncsn2)cc1.C12CCCN1C2=O C(c1ccccc1)=CCNC1CCC(CCNC(c2ccc(C(N)=O)[nH]2)=O)C1 N1(CC(=O)N(C(CCNC(C(C=C)C)=O)C)C)CCC(C)(C)C1 C=CCC(CNC(=O)CC=CC(C)(C)C)C(=O)NC(c1nnc(O)o1)C c1(C(=O)NCCN(C(=O)C(C)(C)C(=O)NC)CC)ccc(OC)c2ccsc12 C#Cc1cccc(C(=O)NC2(CC)CCCN(C(=O)CN(C)C(C)=O)C2)c1 c1(OCCNC(C(=O)N(C)CCc2ccccc2)=O)ccc(C#N)cc1 Cc1cccc(Cn2nc(C3CC3)nc2-c2nnn(C)n2)n1 C(=O)(CS(=O)(=O)Cc1ccc(Cl)s1)N(CCCN(C(COCCC#C)=O)C)C c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2C2CC2)ccc(C(C)C)c(F)c1 CC(C)(C)CCC(=O)N1CCC(C(=O)NCc2ncon2)C1 CCC(CN(C)C)CC(=O)NCC(C1CCCCN1C(C1CCCC1)=O)(C)C CC(C)CC(CNC(=O)CC1CCC=CCC1)C(=O)NC1C2CCCCC12 CC(CC(=O)N(C1CS(=O)(=O)C1(C)C)C)C(C)(C)NC(=O)CN1CC2CC2C1 c1(NC2CC3CNC2C3)nc(Cl)c2c(ccn2C(=O)C(CC(Cl)Cl)C)n1.C(C)(C)C C1(CNC(=O)COC2CCOC2)CCCCN(C(c2cn3c(n2)CCC3)=O)C1 c1(C(=O)NC(CC(C)NC(C(C)SCCCC)=O)C)cnn(CCO)c1N C1(C(=O)NC(C)CN(C)C(C2CCC(O)CC2)=O)CCCC2(C1)CC2(F)F CC(CC1CCCO1)C(=O)NCCCN(C(=O)CCSC1CCCC1)CCO CCCC(CNC(=O)C1=COCCC1)C(=O)NOCC1CCOC1 c1(C(=O)NC(CNC(CCc2c(C(=O)OC)nco2)=O)C)ncnc2cc[nH]c12 c1(OC)cncc(C(=O)NCC2(O)CCN(C(=O)CCc3nc(C)cs3)C2)c1 N1(CC(=O)Nc2cnccn2)CCN(C(=O)CCC2OCCO2)C2COCC12 c1(C(=O)OC)ccc(NCC(=O)NC2CC2NC(c2cnc(O)n2C)=O)cc1 N#Cc1ccc(CN2CC(O)CC2C(=O)Nc2cccc(Cl)c2F)c(F)c1 C1(C(N2CCCC(NC(c3cn(C)c(=O)n3C)=O)C2)=O)CCCC2CCCCC12 Cc1c(NCC2(CC(N)=O)CC2)ncnc1N1CCOC(c2cccc(Cl)c2)C1 C(C)(C)(CCCCNC(=O)C(O)C1CC1)OC(C)=O.N12CCCC1CC2=O c1(C(=O)NC2(CN(C(c3c(SCC)cncc3)=O)C)CC2)ccc2nncn2c1 CCCCC(O)C(=O)N(CC(C)(C)CN(CC)CC)C.C(=O)(C(C)(C)CSC)N CCCCC(CNC(=O)C=C(C)c1ccsc1)NC(c1ccc(COC)cn1)=O C1(C(=O)NC2CCN(C(C3(CC=C)CC=CC3)=O)C2C)CCCC(C)C1C C1(C)(C(N2CCCC(NC(C3(C)CC(F)(F)C3)=O)CC2)=O)CCCCC1(F)F C(C(C(=O)NC1CCOCC12CCC2)C(C)(C)C)NC(C(C=C)CC)=O Cc1c(C(=O)NC2CN(C(c3cnsn3)=O)CC2F)nn2ccccc12 c1(CCC(N2CCC(C)(NC(C(CC)C)=O)CC2)=O)ccc2c(c1)CCO2 c1(OC)cccc(S(=O)(=O)N2CC(CC(=O)Nc3ccc([N+](=O)[O-])cc3I)C2)c1 Cc1cnc2c(C(=O)NC3COCCN(C(C4(O)COC4)=O)C3)cnn2c1 CC(C)C(CO)C(=O)N1CC(F)CC1CNC(=O)CCC1CCOC1 N1(C(CN2CC(=O)NCC2)=O)CC2CCC1C2NC(c1sc(F)cc1Cl)=O N1(C(=O)OC(C)(C)C)CCCC(CCCCNC23CC4CC2C3C4)C1 O=C(C1=C(F)CN(C(c2ccc(Cl)cc2)=O)CC1)NCCC1(O)CCC1 c1(N(CCC#N)C)nc2cccc(F)c2c(=NC2CN(c3cccnc3)C2)[nH]1 c1(C(=O)NC2(C)CCN(C(c3cc(OC)no3)=O)C2)cnc2ncc(Cl)cn12 C1(c2cn(C)nn2)(C(=O)NCCC2(NC(C3CCCS3)=O)CCC2)CCCCC1 N1(C(C=CC=CC)=O)CC(C)CN(C(=O)Cn2nc(Cl)ccc2=O)CC1C C1(C(=O)NCC2C3CN(C(=O)Cc4cc[nH]c4)CC23)CCOC2(CCCC2)C1 C1(C(=O)NCC2(CC=C)CCOC2)CCCCC1NC(=O)C(O)CN(C)C c1(NC(c2c(OC)cccn2)C)ccc(S(=O)(=O)N2CCCCC2C)cc1Cl C(=O)(CC(C)C(C)(C)C)N1CCC(C(C(=O)NCc2cc(C)sc2C)(C)C)C1 c1(OC)ccc(C(c2nnnn2C2CC2)NCC2CC(=O)N(C)C2=O)c(F)c1 N1(C(c2c(C)n(C)cc2)=O)CCC(CNC(c2ccnn2CC2CC2)=O)C12CC2 C(C)(C)(CC(=O)NCCc1cn(CC2CCOC2=O)nn1)OC N(C1CCc2cc(CNC(=O)CCn3ccnc3C)ccc21)C(C(F)OC)=O c1(CC)cc(NC(COC)CC)n2nccc2n1 c1(C(N2C(CN(C(C(CC(C)C)O)=O)C)CCCC2)=O)ccc2nncn2c1 c1(C(=O)NC2(CC=C)CN(C(=O)CNC(C)=O)C2)cc(N)ccc1O C1(NC(c2c(CC=C)cccc2)=O)CN(C(=O)CCC(=O)N(C)C)CC2(CC2)C1 C1(C(N2CC(CC(C(N3CCN(C(C)C)CC3)=O)F)C2)=O)CCC(=O)N(C)C1 c1(C(N2CC(C)(NC(C=CC(=O)OCCCC)=O)C2)=O)n[nH]c(C)c1[N+](=O)[O-] c1(C(N2CC3(CC(O)C(O)CO3)C2)=O)cc(O)nc2c1CN(C1CC1)CC2 CN1CCC(NC(=O)CCC(N)=O)C12CCCN(C(c1c[nH]cc(F)c1=O)=O)C2 c1(CC(=O)NC(c2ccccc2)CNC(c2c(C)noc2)=O)ccc(F)c(F)c1 n1(CC(C)OC)cc(C2CCC2)nn1.C(C(=O)N)CCN(CC)CC.C1(=O)CN1 c1(OC)c(F)cc(C(=O)NC2CC3CC2CN3C(c2ccc(O)cn2)=O)cc1Cl c1(C(=O)NC2CC(NC(CC(C=C)C)=O)C2)cc(=O)n(C)c2ccccc12 C1(C(=O)OC)CN(N2CCC3(CC2)COC3C)CC(C)O1 C1(O)CCC(C(=O)NC)CC1.N1(CC)CCN(CCOCC)CC1.C12(CC1)C(=O)NC2 c1(OC)cccc(C(=O)NC2CCN(C(=O)COc3ccon3)CC2O)c1OC N#Cc1csc(C(=O)NCCCNCC2(Cc3ccccc3)COC2)c1 C=CC(C)(C)CC(=O)NC(C1CCOC1)CNC(c1ccc(C(F)F)cn1)=O C1(NC(c2cccc(OC)c2C)=O)COC2(CCCN(C(=O)C(F)OC)C2)C1 c1(C(=O)Nc2nnc(CN(C)C)s2)c(N)cc(F)cc1Cl C1(=CCNC(=O)CCc2nccs2)CCN(c2cc(-c3ccccc3)ncn2)CC1 C1(NC(c2c[nH]cc(F)c2=O)=O)CCN(C(=O)Cn2ccc(O)nc2=O)CC1O C(N=c1[nH]cnc2c(F)cccc12)C1C(NC(c2cncc(NC)c2)=O)CCC1 c1(C(=O)NCCCOC2CCN(C(C3CCC3F)=O)CC2)ccc(F)c(Cl)c1F C12C3CCC1CN(C3)C(=O)c1cc(ncc1)C(=O)NC2.c1(C(C)(C)C)ccco1 C1(C(=O)NCC2CC(F)(F)C2)CCCN(C(c2sc(N3CCCC3)nc2Cl)=O)C1 C1(CC(=O)N(CC(=C)C)C2CC2)CN(C(C2CN(C3COC3)C2)=O)CC12CC2 Cc1ccc(CCC(=O)N2CCC2C(=O)Nc2cncs2)c(C)c1 c1(C(=O)NC2CC(NC(c3cnc(C4CC4)s3)=O)C2)coc2c1C(=O)NCCC2 CC1(C(=O)NCCCCC(=O)NC2(CO)CC(F)C2)CC(F)(F)C1 CCC(O)C(F)(F)C(=O)NCC1CC1NC(=O)C(=O)N=S(C)(C)=O Cc1nc(C)c(CCC(=O)NC2CCC(NC(=O)CN=S(C)(C)=O)CC2)c(O)n1 CC1C(NC(C2CCC=CCC2)=O)CCCN1C(=O)C1=NOC(C(C)(C)C)C1 CCC(CC1CCCC1)C(=O)N(C1CCCC1)C N1(C(=O)Nc2cc(C#C)cc(N)c2)CC(C2CCC2)CCC1C Cc1ccc(C(=O)NC2CC(CCNC(=O)C(C)c3cccs3)C2)c(C)c1 C1(N(C(c2cncc(NC)c2)=O)C)CCCN(C(C2(C(F)(F)F)CCO2)=O)CC1 c1(C(=O)NCC2(NC(=O)CC3COC(=O)C3)CCCC2)cc2nc(=O)ccn2[nH]1 c1(C(N2CC3C(COC)(C3)C2)=O)cc(-c2ccc(-c3cccs3)s2)cc(F)c1 c1(OCC)cccc(C(=O)NC2CCCC(NC(=O)Cc3ccoc3)CC2)c1N CC#CCCCC(C)(c1nnnn1CC1CCOCC1)NCCC1C=CCC1 C1(C(=O)NC(CCOC)CNC(=O)CSc2nnnn2C2CC2)NC(=O)OC1(C)C C1(NC(C2(C)CC2(Cl)Cl)=O)CN(C(=O)COC2CCC2)Cc2nccn2C1 C1(N(C(c2ncc(C)nc2)=O)C)CN(C(=O)CC2=CCCC2)CCC1O N1(C(C2N(C(=O)OC)CC(F)(F)C2)=O)CC2CCC(C1CO)N2C(C1CC1F)=O C1(NC(CCCSC)=O)CCN(C(=O)C(C)NC(=O)COC(F)F)CC1C(N)=O c1(C(=O)NC2CCCC2NC(C2CC3(C2)CC3F)=O)noc2c1COCC2 N1(C(C2(C(CC)=O)CC2)=O)CCOC(c2cn(-c3ncc(C)s3)nn2)C1 CN1C(=O)CCC1(C)CNC(=O)CC(C)(C)N(C(=O)C=C1CCCCC1)C N12CCC3(CC(C3)C(C3CCC3)CC1=O)C2.N1(C(C(=O)N)=O)CCCC(C)C1.CO n1(CC)nnc2cc(C(=O)NC3CC3NC(=O)C(=O)NCC)ccc12 c1(C(N2C(C(C)NC(c3scc(C)c3)=O)CCC2)=O)cccc(C)c1O N1(C(CCc2cncc(C)c2)=O)CC2(COC(CNC(c3cscn3)=O)C2)C1 c1(NC(C2CCCN(C(C(C)=C3CC3)=O)CC2)=O)cc(C)cc(C#N)c1 CC(CC(=O)NC1CCCC1CNC(=O)CC(C)(C)C(F)F)C(F)(F)F c1(COC)ncc(C(=O)NCC2CCC(NC(C3(C#N)CC3(C)C)=O)C2)c(O)n1 C1(NC(CCCC2(NC(c3c(CC)c[nH]c3)=O)CCC2)=O)COCCOC1 Cc1ccccc1S(=O)(=O)CC(=O)NC1CCCCCN(C(C2CC(F)C2)=O)C1 c1(C(=O)NC(CC)CNC(c2cnc(COC)s2)=O)c(C)ccnc1O Cc1cnc(C(=O)NC2CCCC2CNC(=O)Cc2ncoc2C)cn1 C1(CC)(NC(C2CCCC2C(F)F)=O)CCCN(C(c2cnc(O)c(C)c2)=O)C1 c1(C(=O)NC2CC(NC(c3cccc(O)c3F)=O)C2)cc(F)cc2ccoc12 C(c1nc2ccccc2o1)=CC(=O)NCC=CCNC(=O)CC1CCCC1O c1(C(=O)NC(C(=O)NCC(CC)CC)C(C)C)ccc(C)c(C#N)c1 N1(C(C2(C=C)CCC2)=O)CC(CNC(c2ccc(CO)nc2)=O)C(C)C1 c1(C2(N)CC2)ccccc1.c1(C(C(=O)N2CC(F)C2)O)ccccc1 C1(F)(CNC(C2Cc3nncn3C2)=O)CCCN(C(=O)CN2CSCC2=O)C1 C=CCC(C)(C)CC(=O)NC1COC2(CNC(c3ccc(O)cc3)=O)CC1C2 Cc1cc(C)c(NC(C2CCN2CC(=O)Nc2ccc(Br)cc2)=O)s1 c1(NC(C2CCC(NC(=O)Nc3ncc(F)cc3Cl)C2)=O)nc(Cl)c(Br)cc1I CC1CCC(C)(C(=O)NCC2CC2CN(C(=O)CN(C(=O)C(C)C)C)C2CC2)CC1 C1(NC(Cc2cccc(OCC)c2)=O)CN(C(=O)C(C)(C)F)CCC1O CC1CCc2onc(C(N3CC(CNC(c4cccc(S(C)=O)c4)=O)C3)=O)c2C1 c1(CC)cc(C(N2CCC(CO)(NC(c3cc(OC)ncn3)=O)C2)=O)ccc1C C1(N(C(CC(C)SC)=O)C)CCCCN(C(=O)CC(=O)OC(C)(C)C)C1 c1(C(=O)NCCOCCNC(c2cnc(C(F)F)s2)=O)ccc(F)o1 CC(CCC(=O)NCCOCCN(C)C(c1ccco1)=O)S(C)(=O)=O c1(C(C)C)nccn1CC(=O)NCC1CC1NC(C1(CCF)CC1)=O N1(C(c2ccc(OC)nn2)=O)CCCC(NC(C2CCS(=O)(=O)CC2)=O)C(F)C1 Cc1cc(C(=O)NCC2(F)CC(CNC(=O)CC3CC(O)C3(C)C)C2)c(C)[nH]1 C1(CC(=O)NC(C2CCCN2C(=O)CSCC(N)=O)C)C(C)(C)C1(C)C N1(C(CN(C(=O)CC2CCCOC2)C(C)C)=O)CCC(C(F)F)C1 c1(C(CNC(C(C=C)O)=O)NC(c2cccc(OC)n2)=O)cccc(C)c1 C1(CC)C(NC(=O)CO)CCCN1C(c1nnn(C2CCOC2)c1C)=O Cc1cc(C(N2CC(O)CC2C(N2CC(CC3CC3)C2)=O)=O)c(C)cn1 Cc1c(C(=O)NC2CC(NC(C3(CF)COC3)=O)C23CCC3)cccc1O Cc1cc(C(=O)N(C)CCn2cccn2)[nH]c1C c1(C(=O)NCC2(F)CCC(NC(C(CC)(C)CO)=O)C2)cc(OC)c(N)cc1F c1(C2(C)COCCO2)ccc(-c2ccc(NCc3csc(C(F)(F)F)n3)s2)cc1 N1(C(c2ccc(OCC)cc2)=O)CCC(C(F)(F)F)C(NC(=O)CC2CSC2)C1 c1(C(N2CC(C3CC3)C2)=O)cc2occ(C)c2[nH]1.CCCCCOCC.C1C(=O)N1 c1(C(=O)NCC2N(C(C(C)OCC)=O)CCC2C)ccc2c(c1)SCC(=O)N2 c1(C(=O)NC2CN(C(C(C)SC(F)(F)F)=O)CC(F)C2)cc2nn[nH]c2cc1F C1(C(C)(C)C)C(=O)N1.C(CC(=O)NCC1(CF)CCC1)NC(=O)NC CC1CN(C(=O)CNC(C2CCCN2C(=O)OC(C)(C)C)=O)CC(C)(C)CO1 Cc1nnc2n1CCN(C(=O)C(N1CCNC(C(F)F)C1)=O)C2C CN1CCCC(C)(C(=O)N(CCNC(c2cc(Cl)ncc2N)=O)CC2CC2)C1 C1(C(=O)NCC2(CN(C(=O)CCc3cncs3)C)CC2)CCCC(O)C1 C1(C(N(CCN(C(C2CC(OC)C2)=O)C)C(C)C)=O)CC(C)(C)CCO1 c1(C(N2CCC(NC(C3C(C=C)OCC3)=O)C(O)C2)=O)ccc2c(c1)CCOC2 N1(C(C(CC)=O)=O)CCC2C(CCN2C(c2n[nH]c3cccnc23)=O)C1 N1(C(C2C(NC(=O)OC(C)(C)C)C2(C)C)=O)CC=CCC12CCCCC2 c1(C(N2CC(C(C)NC(COC)=O)OCC2)=O)c[nH]c2cccc(C)c12 Cc1cc(Cl)c(Cl)cc1C(=O)N(CCCCCNC(C1COCCO1)=O)C N1(C(C(CC)N2CCCC2=O)=O)CCC(O)(CO)CC1 c1(C(=O)NC2CC(NC(C3C(C)(C)OC(=O)C3)=O)C2)cc2cccnc2cc1F C(=O)(C(C)CC(C)(C)C)NCC(CNC(CCN(CCCCOCC)C)=O)O N1(C(C2CC(SC)C2)=O)CCCCC2(CCN(C(c3ccnc(C)c3)=O)C2)C1 c1(C(=O)OCC)cc(NC(=O)NC2CCCC(C(N)=O)C2)cc(F)c1 C=CC1CN(C(=O)C(C)(CNC(=O)CCCNC(C)=O)CC)CCO1 C(=O)(CC(C)C(F)(F)F)N1CC(OC)C(C(=O)N(C2CCC(CO)CC2)C)C1 c1(CC(=O)N(CCC(=O)N(C)CCOCCO)C)cc(F)ccc1F C12(C(=O)NC(C)CCN(C(=O)CN(C)S(N)(=O)=O)C)CCC(O)(CC1)CC2 c1(C(=O)NCC(CCNC(CSCC#C)=O)OC)cc(OC)cnc1F C1(C(=O)NCCOC)CCC(C)CN1C(=O)C(=Cc1ccccc1)C Cc1nc2ccccn2c1NC(c1ccnc(-c2ccn3ccnc3c2)c1)=O N(C(=NCCC(C)=O)N1CCC(O)C1)CC(=O)N(CC(F)(F)F)CC.C(C(C)C)OC c1(CC)cc(F)c(C(=O)NCC2COCC2NC(c2[nH]cnc2C)=O)c(F)c1 c1(CCC(=O)N(CC(c2ccccc2)NC(CCCC)=O)CC)ccc(C)cc1 C1(CC=C)(NC(=O)C(C)CCCC)CCN(C(C)=O)CC1 c1(N2C(C(C)NC(C3(C(N)=O)CC3)=O)CCC2)ncnc(-c2ccccc2)n1 C1(C(=O)NC2(CNC(c3cnc(C(C)C)[nH]3)=O)CCC2)Cc2ccccc2C1C C1(CNC(C2N(C(=O)NC)CCC2)=O)C(C)CCCN1C(c1ocnc1C)=O c1(C(=O)NC(C2CCN(C(=O)C3=NOCC3)C2)C)n[nH]c2cc(Br)ccc12 c1(C(=O)NCC(CC)NC(c2cnnc(Cl)c2)=O)cc([N+](=O)[O-])cn1C C(=O)(C1CC(=O)Nc2ncccc21)N1CCC(C(C)NC(c2ccco2)=O)CC1 CCC(C)(C)C(O)C(=O)NC1CCN(C(c2cc(C(F)F)ccc2F)=O)C1 c1(C(=O)OC)ccn(CC(F)(C#N)C(C)C)c(=O)c1 CC1CC(C)CCN(C(=O)CCC2(NC(c3sccc3C#N)=O)CCCC2)C1 N1(C(C2C(OCC)C2C)=O)CCC(NC(C2(C)CCCS2)=O)C1c1ccccc1 C(=O)(C1=CN=C2N=CNN2C1)N1CCCC(C(C)NC(CC(C=C)(C)C)=O)C1 c1(C(=O)NC2C(NC(c3c(C)nsc3)=O)COC2)ccc2c(c1)CN(C)C2 c1(C(=O)NC(C(=O)NCC2C(C(=O)OC)C2)c2ccco2)cccc2ccoc12 C12(NC(C(C)(C)c3ccno3)=O)CC1CN(C(c1ccc(C(N)=O)s1)=O)C2 C1(NC(CCc2cc(C)[nH]n2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC2(CC2)C1 CCC(CC(=O)NCCC1(NC(=O)C(C)(C)c2cscn2)CCCC1)SC c1(C(N2CCC(OCCCNC(CC(C)SC)=O)CC2)=O)cccc(=O)n1C C1(NC(C(CCC)N(C)C)=O)CS(=O)(=O)C12CCN(C(C1(CF)CC1)=O)CC2 C=CC1CCCCN1C(C1CCCC(C)C1)=O c1(C(=O)OC)cc(Nc2ccc(C3CC3C)o2)ccc1Cl.C12CCCCN1C2=O N1(C(CC=CCC)=O)CCC(C)(C)C(CNC(=O)C(CC)SCC)C1 C1(NC(CC2(CC=C)CCCC2)=O)CCC12CN(C(=O)C(c1cnn(C)c1)O)C2 c1(C(C)=O)cc(N2CC3CC(NC(=O)C=CC4CCC4)CC3C2)ccc1[N+](=O)[O-] C1(c2nc(C(C)(C)OCC3CCN(C)CC3)on2)CCOCC1(C)C c1(C(N2CC(NC(C(CC)COC)=O)C(O)C2)=O)cnc(C)nc1C(C)C Cc1csc(CN(C(=O)CC2C(NC(=O)CC(C)n3cccn3)CC2O)C)n1 Cc1cc(C(=O)NCC2CCCN2C(c2cc(=O)n(C)o2)=O)oc1C C1(C(C)(C)NC(=O)C(C2CC2)C2CC2)CCN(C(C2(CO)CCCO2)=O)CC1 C1(NC(c2c(C)[nH]nc2Br)=O)CN(C(C2OCCN(C)C2=O)=O)CC2CC12 C1(C(N(C2(CC(=O)N(CC(C)SC)C)CC2)C)=O)CCCCCN1C C1(CNC(CC(C)(C)NC(C(C)C2CCOC2)=O)=O)OCCCC1(C)C C1(CNC(C2CC(C)(F)C2)=O)CC2(CCN(c3ncnc4[nH]cnc34)C2)CO1 C1(n2cc(C3CCOC3)nn2)(C(=O)NC(C)Cc2nccn2C)CCOCC1 C(=O)(C1=CCCC1C)N(CCC(=O)N(C)Cc1ncc(C)o1)C1CC1 CC(C(=O)NCC(O)CCNC(=O)C(c1cc(F)cc(Cl)c1)=O)C(C)(F)F N1(C(C=CC=CC)=O)CCC(NC(=O)C(C)OCCOC)C12CCCC2 C1(C(N)=O)C2C=CC2CN1c1ccncn1 CCCC(C(F)(F)F)NC(C1(F)CCN(C(C2SCC=C2C)=O)CC1)=O C1(C2CN(C(=O)C=C3CCCC3)C2)(N(C(CC(C)(C)C)=O)C2CC2)CC1 Cc1[nH]nc(CO)c1C(N1CCC1C(N1CC2CC2C1)=O)=O c1(C(=O)NCCC(CC)(C)NC(c2nnsc2C)=O)ccc(OC)c(C)c1 N1(C(c2cn(CC(=O)OC)nn2)=O)CCC(NC(C2CCCC2)=O)C(C)C1 c1(CCC)nnc(S)n1CC(N1CCC(C)(CNC(=O)CCc2cscn2)C1)=O C(=O)(CCCCC(C)C(C)C)NCCN(C(c1cnc(OC)nc1)=O)C(C)C N1(C(C2(C(C)C)COC2)=O)CC2(C1)CN(C(=O)COc1ccc(F)cn1)C2 c1(CC)nn(C)c(CC(=O)NCCN(CC(C)O)C(c2ccsc2Cl)=O)c1Cl c1(C(N(CCC)CCNC(c2cnn(C(F)F)c2)=O)=O)cc(COC)cn1C c1(C(N(CCCCNC(c2cc(OC)cc(F)c2)=O)C)=O)cc(O)cc(N)c1Cl CC(CN(C)C)CCC(=O)N1CC(C)(C)CC1CNC(C1CC12CCSCC2)=O C(C(C)C)(C(O)C(=O)N1CC2(C1)CN(C(=O)Nc1cc(C)ccc1Cl)C2)OC C1(C(N2CCC(C=C)CC2)=O)CC12CCN(C(=O)CSCCC)CC2 C=C(Cl)CC(C(=O)N(CCN=[N+]=[N-])CC)NC(c1cc(F)ccc1O)=O c1(OC)cccc(C(N2CCC(NC(c3c(C)ncn3C)=O)CC2C)=O)c1C N1(C(CCC(=O)NCCCC)=O)CC(O)CC1CC(N1CC2CC2(CO)C1)=O C1(NC(C2C(N(C3CCCNC3=O)CC)CCC2)=O)CCN(CCC2CC2)CC1 CCC(C)(CN=C(NC(c1ccc(C(C)C)cc1)C)NC1CCCCC1)OC c1(CN2C3(CN(C(=O)Cc4ccc(O)cc4)C3)CC2)ccc(O)c(F)c1F Cc1ccc(Cl)c(C(=O)NCC(C2CC2)NC(c2ccc(OC(C)C)cc2)=O)c1 C=CC(C)(C)CC(=O)N1CCC(O)(CCNC(=O)C(C)(CC)OC)C1 Cc1ncc2n1CCN(C(C1(CCNC(c3cnc4n3CCC4)=O)CC1)=O)C2 Cc1nn(C)cc1C#CC(=O)N(CCCn1cc(CC(C)(C)O)nn1)C C1(CNC(CSCCOC)=O)CN(C(c2ncncc2C)=O)CC1O CC1(C)OC2(C(=O)NC3CCC3NC(c3c[nH]c4nccc-4c3)=O)CCC1CC2 CCC(CCOCO)NC(=O)C=CC(N1CCC(OCCOC)C1)=O c1(CNC(C(Cc2ccco2)NC(CSCC(N)=O)=O)=O)cncc(Cl)c1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2CCN(C(=O)C(C)(C)SC)CC2C1 C(C)(C)(C(C)CC(=O)N1CC(N2CCCC2=O)C1)NC(C(C)SC(C)C)=O C1(NC(C(C(C)C)OCC)=O)CCCC12CN(c1nnc(CC(F)(F)F)s1)C2 c1cnn2ccn(C)c12.CCC1(CC)CCNC(=O)C2(COC2)C(=O)N1.COC C=CC1(NC(c2ccccn2)c2nnnn2C2CCC2)COC1 c1(NC2CCC(CC)C2)cc(C)c(S(=O)(=O)N(C)CCCC2CCCCC2)cn1 Nc1c(C2CC3(CC(CNC(c4cnoc4)=O)C3)C2)ccc(F)c1F Cc1cc(N)c(C(=O)NCC(C)NC(C2CCCN2C)=O)nc1C N1(C(c2ccc(CO)cc2)C(=O)NCC=C)CC2(CCCCC2)CC1C O=C(CC1NC(=O)NC1=O)NNC(=O)c1ccc(C(F)(F)CF)cc1 c1(C(=O)NCC(CO)NC(Cc2c(C)ccs2)=O)ccc2c(c1)COCCN2 Cc1cnncc1C(N1CCCC(NC(c2ccc(CN(C)C)o2)=O)C1)=O CN1CC(C)(C(=O)NC2C=CCCC2C(N2CC(F)(F)C2)=O)CC1=O c1(NC(CCn2ccc(C)n2)=O)ccc(NC(=O)Cc2cocn2)c(C)c1 CC1CC(NC(=O)C=CCO)CN1C(c1cnc(S)n1C)=O C1(C(=O)NCCN(C(CCCOC(C)C)=O)CC(C)O)CC2CCCCC12 c1(C(=O)NC(CC)CNC(c2nncs2)=O)cccc(-n2cc(C#N)cn2)c1 C(CN=C(NCC(C)(C)CC(F)F)NCc1cccc(C(C)C)n1)OC c1(C(N(C(C)C(=O)N(CC(C)C(C)C)C)CCC)=O)cc(NC)ccn1 c1(CN2CCN(C(C(=O)NCCCSC)C)CC2)cc(OC)c(OC)cc1C N1(C(C(CC)CO)=O)CCCC(C2CC2NC(c2csc(S)n2)=O)C1 CCC(C)CC(C(=O)NCCC(C)C(=O)OC)NC(=O)CC1CCOC1C c1(OC)cc(C(=O)N(C2CC(NC(=O)C(N3CCCC3)C3CC3)C2)C)on1 C1(CNC(CC2(C=C)CC2)=O)CC(NC(=O)CCCc2ccccn2)C1(C)C C1(C(CO)N(C(=O)CSc2ncc[nH]2)C)CCN(C(=O)OC(C)(C)C)CC1 CCC(O)CC(=O)NCCCC(=O)NCCc1cccnc1F C1(NC(c2cnco2)=O)CC2C1CCN2C(c1cnc2n1CCC2)=O c1(C(N2CCC(CN(C)C(c3cc(C(=O)N(C)C)[nH]n3)=O)C2)=O)cnc(O)c(F)c1 CCS(=O)(=O)c1ccc(F)c(C(=O)NC23CC2CN(C(=O)C2=CCCC2)C3)c1 N1(C(CCCN(C(C2C(C)CCCC2)=O)C)=O)CCC2CCCC2CC1 C1(CCNC(C(C)Cc2ccnn2C)=O)CC(F)(F)CN1C(c1cncn1C)=O CCC(C)(O)C(=O)N(CCc1cn(-c2ccnc(C(=O)O)c2)nn1)CC C12(Cn3cc(NC(C(CSC)C(N4CCCC4)C)=O)nn3)CC3CC(CC1C3)C2 C1(C(C)C)CC(CC(=O)N(C2CCN(C(=O)CC=C(Cl)Cl)CC2)CCO)CCO1 C(N=c1[nH]c2cccc(F)c2s1)C1N(C(C2CCCS2)=O)CCCC1 c1(C(=O)NC2CN(C(c3c(CC)nc[nH]3)=O)C(C)CC2)nc2ncccn2n1 c1(C(=O)OC)c(C(=O)NC(CNC(C2CN(C(C)C)C2)=O)CO)n[nH]c1C C1(CNC(c2n(CC#C)ccc2)=O)CN(C(=O)C2CC2)CC1C(F)(F)F c1(C(=O)NC2C=CCN(C(C(C(C)C)NC(N)=O)=O)C2)ccc(F)c(F)c1 c1(C(=O)NCC2C(NC(C(C)N3CCC3)=O)C2)n[nH]c2c1CCOC2 c1(CCSC)cccnc1NC(c1cc(C)sc1N(C)C)=O c1(C(=O)NCC(CNC(=O)COCc2ccncc2)F)ccc(F)c(O)c1F C1(N(C(Cc2ccc(C)o2)=O)C)CN(C(C2CC(F)(F)C2(C)C)=O)CC12CC2 C1(C(=O)NC2CCOCC2NC(c2sc(CO)nc2C)=O)(COC)CCOCC1 Cc1ccccc1-n1ccc(C(=O)NC(CNC(c2cnn(C)n2)=O)C(C)C)n1 C#CCCC(O)C(=O)NCc1ccc(CNC(=O)C(C)S(N)(=O)=O)cc1 c1(C(N(C2CCN(C(c3cc(F)n[nH]3)=O)C2)C)=O)cnc(C2OCCO2)s1 C1(NC(C2(C)CC2(F)F)=O)CN(C(c2nonc2N)=O)CC1c1ccccc1 Cn1nc(C(=O)NC2CC(O)(CNC(=O)CCC(C)(C)F)C2)cc1C#N c1(C(N2C(CNC(C3NC(=O)C(F)C3)=O)CCC2)=O)ccc(=O)n(CCF)n1 Cc1ccc(N)c(C(=O)NCc2ccc(CNC(C3CC3(F)F)=O)cc2F)c1F n1(CCCC)nnnc1C(c1cncs1)NCC(C1CCC1)OC c1(OC)ccc(F)c(C(N2CCC(NC(c3ccn(CCO)c3C)=O)C2)=O)c1N c1(C(=O)NC2C(NC(C(C)(CO)NC(C)=O)=O)COCC2)n[nH]c2c1CCCC2 c1(C(=O)NC(c2cc[nH]n2)CNC(=O)CC2CCOC2)cc(F)c[nH]1 c1(C(=O)NC(c2cn(-c3nonc3C(=O)O)nn2)C)ccnc2c1cnn2C c1(CC(N2C3C(NC(Cc4c(C)nc[nH]4)=O)C(C3)C2)=O)cn2cc(F)ccc2n1 c1(NC(C2(C)CN(C(CCn3ccc(C)n3)=O)C2)=O)cc(F)cc(Br)c1 C1(OC)CCC2(CCN(C(=O)NC(C3CCCO3)C3CCCC3)C2)C1 n1(CC)cccc1NC(=O)Cc1cn(CC2CN(C(c3cocc3C)=O)C2)nn1 C1(CC)CCN(C(C2CC2CC)=O)C1CNC(=O)CSCC1CCCO1 C(C(C)CCCO)NC(C#CCN(C(Cc1nc(C)oc1)=O)C)=O c1(C(N2CCOCC(NC(C(C)S(N)(=O)=O)=O)C2)=O)ccc2c(c1)CCO2 C(CCCSC)(C(=O)NC)N1CCN(C(c2ccccc2C)C(=O)NCC)CC1 N1(C(C(C(C)O)(F)F)=O)CCC2(CCC2)C(NC(=O)CCn2ccccc2=O)C1 N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)CCSc2ccoc2)C(CO)CC1 N1(C(c2c(CC)ocn2)=O)CCC(CNC(c2[nH]c(=N)ccc2C)=O)C(C)C1 c1(C(=O)NC(CN(C(=O)CCCF)C)(CO)CO)cnc2n(c1=O)CCS2 N1(C(=O)OC(C)(C)C)CCC(C2CC2)CC1.C1(=O)C(Cc2cncs2)C(=O)N1 Cc1cccc(-c2ccc(C(=O)NCCN(C)C3CC3)cc2)c1 C12(NC(c3ccc(C)nn3)=O)CCC(C(=O)NCC(O)C3CC3)(CC1)C2 C=C(C)C(CC(=O)N(CCCNC(=O)COCc1ccoc1)C)OCC N1(C(CCC(C)OC)=O)CCCCC(NC(=O)C=Cc2cnn(C)c2)C1 c1(C(=O)NC2CC(NC(Cc3ccc(C)c(O)c3)=O)C2)cc2sc(Cl)cc2s1 C1(C(=O)NOCC2CCOC2)CCCCN(C(C2CN3CCC2C3)=O)C1 C1(CNC(CC(C)C)=O)CC2COCC2N1C(C1CCOC1C(C)C)=O C(=O)(C(F)CC(C)(C)NC(C1CC2C=CC1C2)=O)N(C1CCN(C)CC1)C N1(C(C2(COC)CC=CC2)=O)CCCC2(CCC(NC(=O)CO)C2)C1 N1(C(CCC)=O)CCN(CCNC(C2CCC(=O)N2C)=O)C2(CCC2)C1 C1(CNC(CCN(C(CCC)C)C)=O)(NC(=O)CCOC(C)C)CCCCC1 c1(CC)cccc(NC(C2(O)CN(CC(O)CC3CCCC3)C2)=O)c1 c1(C(=O)NCC2N(C(C3C(C#N)C3)=O)CCOC2)cc2cncn2c(O)n1 CCC1=NOC(C(=O)NCCCC2(NC(c3coc(C#N)c3)=O)CC2)C1 c1(C(N(CCC(C)NC(COC(CC)C)=O)C)=O)n[nH]c2c1COCC2 c1(C(N2CC3C(NC(C4C(C(N)=O)C4)=O)(C3)C2)=O)cc2ccc(Cl)cc2c(O)n1 CN1CCCCC(C(N2CCN(C)CC2CNC(=O)CSc2nncs2)=O)C1=O Cc1cc2cccc(C(N3CCCC(N4CCNCC4=O)C3)=O)c2o1 C1(OC)CC(N2CCC2)N(C(CC(C)(C)C2CCCO2)=O)C1 c1(C(N2C3CN(C(C(CC#C)C)=O)C(C3)C2)=O)ccc(S(=O)(=O)CCO)nc1 C1(C(N(CCCN(C(c2cc(C(C)C)on2)=O)C)C)=O)CC(F)(F)C12CCC2 C1(C(=O)NCC(C)(C)NC(=O)CC2CCC(=O)NC2=O)CCCCC(F)(F)C1 C1(CC(N2CCC(C(=O)NCc3ncc(C)cn3)C2)=O)CC=C(C(C)C)CC1 N1(c2nc(C#C)sn2)CCC(CO)C(C2CC2)C1 Cc1sc(C)c(C(=O)N(C)CCNC(C2CCC3CC3CC2)=O)c1Br CC(O)C(C)C(=O)N(CCCCNC(C1(c2ccccc2)CC(F)C1)=O)C Cc1ccc2c(c1F)CN(C(=O)Nc1ccc(C#N)cc1F)CC2 C1(NC(C(C(C)C)n2ncc(C)c2)=O)COC2(CCN(C(=O)C=CCF)CC2)C1 N1(C(C2CC3CCC2C3)C(=O)N(C2CC2)CC2CC2)CCCCCCC1 n1(CCC(N2C3C(NC(CN(C)CC)=O)C(C3)C2)=O)cc([N+](=O)[O-])c(O)nc1=O N1(C(COCCOC)=O)CCC(CNC(c2nc(C)nn2C)=O)CC1 c1(-n2ncc(OC(CC(C)NCC(O)C(F)(F)F)=O)c2)c(F)cccc1F c1(N(CCCC)C(c2cnc(NC)nc2)=O)cc(Cl)c(C)c(CC)c1OC N1(C(C(C=CCCC)O)=O)CCN(C(=O)COc2cncc(Br)c2)CC1CC c1(C(=O)NC2CN(C(c3c(C)nns3)=O)C2)ccc(O)cc1F Cc1cc2sc(C(=O)NC3COCCN(C(=O)Cc4nc(C)c(C)s4)C3)cc2s1 N1(C(C2(C)CSC2)=O)CC2CC(C1)CN(C(=O)C(O)CN1CCOCC1)C2 N1(C(CSCC=C)=O)CC(CNC(c2ccc(Cl)c(C(F)F)c2)=O)CC1(C)C C(CNC(=O)C(C)=C1CCC1)(C(C)C)NC(C1(COC)CCC1)=O C(=O)(C(O)CC(C)(C)C)N(C)CCONC(=O)CC1CC(C)(C)CO1 CC(C(C)C(=O)NCC(F)Br)NC(=O)C=Cc1ccsc1 C1(COC)(NC(c2ccc(C3COC3)cc2)=O)CCN(C(=O)CS(C)(=O)=O)C1 C(=O)(C(CN(C)C)NC(C1C(C)C1C)=O)NCCC N1(C(CCC(C)O)=O)CC2(CC2)CC1CNC(=O)C1=NOC(C2(O)COC2)C1 C(=O)(CC(O)CC(C)C)N1C(CNC(C(CC=C)CC)=O)(COC)CCC1 c1(C(N2CCN(C(C(C)C(C)(F)F)=O)C3C2CC3)=O)ccc2c(c1)OCCC2 c1(CNC(COCC#C)=O)cncc(C(N2CCCC2CC(N)=O)=O)c1 S(=O)(=O)(CCN=c1cccc(S(=O)(=O)N2CC(C)OCCC2C)[nH]1)NC O=C(CCN(C(=O)CCn1ccnn1)CCO)NCC(O)CC1CCC1 Cc1ccc(S(=O)(=O)NCc2cnc3n2CCOCC3)cc1C(=O)N(C)C C1(C(=O)NC(CC(C)C)CNC(=O)C(C)(C)C2CC2)CCCCC12CC2 c1(C(=O)NCC(O)CC(=O)Nc2cnc(F)nc2)cnc(O)c(F)c1 C1(C(N(CC(C)(C)NC(c2cnc(C)nc2)=O)C)=O)COc2ccccc2O1 C1(N(C(=O)CC(F)F)C)C2CN(C(c3cnn(C)c3Cl)=O)CC12 C1(NC(C(COCC)C)=O)CN(C(=O)C(C2CC2)OC)CC2(CCC2)C1 c1(C(N(CCC)CCNC(=O)C2=C(C)CCC2)=O)cccc(P(C)(C)=O)c1 c1(C(=O)N(C(C)CC(=O)N(C2CC3CC3C2)C)C)cc(COC)no1 C1(NC(C2CC(N=[N+]=[N-])CN2C(=O)OC(C)(C)C)=O)CCC2C(CC1)C2(F)F N1(C(CSc2cccc(C#N)c2)=O)CCN(C(=O)C(F)n2ccnc2)CC12CC2 C1(CC2CC2)CCCN(C(=O)CCN(C(CC(CC)C2CC2)=O)CC)CC1 N1(C(C(C)OC)=O)CCC(c2c[nH]c(CNC(=O)C(O)(C3CC3)C3CC3)c2)CC1 CC(C)C(=O)NCCC(C)N(C(=O)CCC1CCCC1)C C#Cc1cccc(C(=O)NCC23CCC(C2)N(C(c2ccccc2C)=O)C3)c1C C(CC1=CCN(C(=O)COc2ccsc2)CC1)NC(C1(COC)CC1)=O Cc1nnc(C(=O)NC2(CNC(c3coc(-c4ccccn4)n3)=O)CCCC2)s1 C1(S(N)(=O)=O)(C(=O)NC(C)(C)CN)CC1.C(C(=O)NCC)SCC#C N1(C(CCCOC(C)=O)=O)CCN(C(c2cc(-c3ccco3)ncn2)=O)C(C)C1 c1(SC)ncc(N)c(C(=O)NC(C2CCCCC2)CNC(=O)C(CO)N(C)C)n1 C12(CNS(CC)(=O)=O)CC1CN(C(c1ccc(-c3sccc3C)cc1)=O)C2 N1(C(C2C(C)OC(C)C2)=O)CC2(CC(S(C)(=O)=O)C2)C1 c1(OC)cc(Br)cc(C)c1NC(=O)C=C1CCN(Cc2cc(Cl)ccn2)CC1 CCCC(CC)CC(=O)NC1CCCN(C(=O)Cn2cnc([N+](=O)[O-])n2)C1 CC1C(C)=NOC2CN(C(C3(C(N)=O)CN(C(=O)OC(C)(C)C)C3)=O)CC12 C1(NC(CC2CCC(C)C2)=O)CCC12CCCN(C(=O)CC(=O)NC1CC1)C2 c1(CC)cc(NC(=O)C(CC2CCC2)NC(C2CC23CC3)=O)ccc1F C1(CCNC(C2CCCN(CCC)C2)=O)CCN(C(=O)C#CC2CC2)CC1(F)F C(=O)(CS(C)(=O)=O)N1CC(CC)(NC(=O)C(O)Cn2cncn2)C1 N1(C(C2(Cl)C(C)(C)C2)=O)CC(C2CN(C(c3cc(NC(N)=O)ccc3Cl)=O)C2)C1 c1(C(=O)NCC2C(C(N(C(C(C)C)C)C)=O)CC2)cnn(C2CCC2)c1 Cc1cccn2cc(C(N3CC(NC(=O)C(c4ccccc4)C)C(F)C3)=O)nc12 C#Cc1ccc(C(N2CC(O)(C(C)NC(c3cnn(CCCC)c3C)=O)C2)=O)o1 c1(OC)cc(F)cc(C(=O)NCC2(OC)CN(C(=O)C(O)c3ccsc3)C2)c1N CCC(C(=O)NCC(C(N1CC(CO)C2(CCC2)C1)=O)C(C)C)C(F)(F)F c1(C(N2CCC(CCNC(c3ccco3)=O)C2)=O)cc(O)nc(O)c1 N1(CCOC)CC(Oc2nc(CC(N3C4CN(C(C)=O)CC34)=O)cs2)CC1=O CC(CS(C)=O)C(=O)N(CCCNC(=O)CCCCN1CCOCC1)C1CC1 Cc1cc(F)cnc1C(N1CCN(C(=O)CC2CCC(C)O2)CC1)=O CC(C)C(C#N)C(=O)NC1(CNC(c2cnc(C(C)(C)C)o2)=O)CCCCC1C C1(C(N2CC(NC(CCSC)=O)C(c3nccn3C)C2)=O)Cc2nccn2C1 C1(C(C)NC(c2cocn2)=O)CCCN1C(c1c[nH]c(-c2ccccc2)c1)=O CC1CN(C(=O)CC2CCN(C(=O)CCN(C)C)C2)CCC1CO N1(C(C(C)(C2(C)CC2)OC)=O)CCOC(C(=O)N(C)CC2C(C)(C)C2(C)C)CC1 C1(C(=O)NC2CCCC23CC3)(CC)CCCN1C(=O)CCn1ccnn1 C(Cc1ccoc1)(C(=O)NCCCC1CCOC1)NC(C1C=CCS1)=O Cc1cnc(C(=O)NC2CCC(NC(C3CC4CCC3O4)=O)CC2)cc1Br C1(NC(C(C(CC)C)NC(=O)CC2CC(OCC)C2)=O)CCC(=O)NC1(C)C c1(C(N(CC(C)NC(=O)C(O)C2CC2)CC)=O)cc2ccccc2c(OC)n1 C1(C(n2cc(C3(N(C)C)CCOC3)nn2)C)CCN(C(c2ccc(F)cc2)=O)CC1 C12C3CCC(C3)C1NS(=O)(=O)CC(=O)NC2=O.C(=O)(C(C1CC1)N(C)C)NC C1(CC(=O)NCCCCNC(c2ncn(CC)c2)=O)CC(OC)C1(C)C C1(OC(CSC(c2ccccc2)C(=O)OC)=O)CCN(C(=O)OC(C)(C)C)CC1 CC(=O)CCCCCc1cccc(NC(=O)C(=O)NC2CC23CC(C(=O)O)C3)c1 c1(C(N2CC(F)CC(NC(Cc3c(C)nn(C)c3)=O)C2)=O)cnc2ncccn12 c1(N2CCCC3(NC(C=CS(C)(=O)=O)=O)C(C2)C3)ncnc2cc(Br)sc12 C(=O)(C1=C(F)CN(C(=O)C(c2ccccc2)C)CC1)NC(C)CC(N)=O CCC(C)C(C(=O)NCC1C2CN(C(=O)C(c3ccccc3C)(C)C)CC12)OC C1(CC(=O)NCC(CC)N(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C)CCCC1O C(=O)(C1=CCCOCC1)NCC(CC(C)C)NC(=O)Cc1ccc2occc2c1 Cn1cnc2nc(=NC(CF)C3CCCC3)[nH]cc12 N1(C(C(C=C)(C)O)=O)CC2(CCCCN(C(c3cnn(CCOC)c3)=O)C2)C1 C12CCN(CC1)N(C)CCc1cn2nn1.C12(C(=O)OC)CCC(OC)C1C2 C=CC(C)(CCN(C)C)C(=O)NCCC1(C)CCN(c2cccc(CSC)c2)C1 C12(NC(C(C)C(F)F)=O)CCC(C1)N(C(c1cc(Cl)cn1C)=O)C2 C(=O)(C(N)CCC(=O)O)C(C)C(N)CCCN C(CC(C)N=c1nc(N2CCC(c3cnn(C)c3)C2)c2ncn(C)c2[nH]1)OC C(C(CC(C)C)C(=O)N1CC2CCCC2C1C(N1CC(O)C12CCOCC2)=O)OC c1(C(=O)NC2(CCNC(CN(C(C)=O)C)=O)CCCC2)cc(C)cc(F)c1N N1(C(c2c(CC)noc2C)=O)CCC2C(C1)CN2C(=O)C(C(C)(C)C)N(C)C c1(C(=O)NC2C(C(N3CCC(C#N)C3)=O)CCCC2)cc2cccnn2c1 N1(C(COC)=O)CCCC(C2(NC(c3sc(S(N)(=O)=O)cc3C)=O)CC2)C1 N1(C(Cc2nc(C)oc2)=O)CCCN(C(=O)CCOC2CCCCC2)C(CO)C1 C(=O)(CC(C)(C)CCCN=[N+]=[N-])N1CC(N(C(=O)CCc2nc(O)n[nH]2)C)C1 O=C(CCC(CF)CF)NC1CC1CNC(c1ccc(C(N)=O)[nH]1)=O c1(CNC(C(CC)=O)=O)ncccc1C(=O)O.C12(C)CCCN1C(=O)CC2 C1(C(N2CCCC(C)C2CN=c2nc[nH]s2)=O)CCCC2CCCN12 CC1=CCC(C(N2CCC(N(C(=O)CN3CCCNC3=O)CCO)C2)=O)CC1 CC1CC(N)CCN1C(c1ccc(=O)n(C)c1)=O C1(C(=O)NCc2cc(Cl)ccn2)CC2CCC1N(C(=O)C1=CC3C=CC1C3)C2 c1(NC(C2CCN(C(c3c(C)ccs3)=O)CC2)C)ncnc2sc([N+](=O)[O-])cc12 C1(CC(=O)NCC(C(C)C)O)CC(C)(C)CN1C(=O)CC(Cl)Cl c1(C(=O)NCCN(CCC)C(C2CCN(C)CC2)=O)cncc2nc(O)[nH]c12 N1(C(CC(C(=C)C)OCC)=O)CCC2(CCC2)C(CNC(C2CSCN2C)=O)C1 c1(NC(=O)NCCNC(C2C(c3nc(C)[nH]n3)C2(C)C)=O)cnn2cnnc2c1 CCCCC(C)C(=O)NC1CCC(NC(=O)C(c2ccccc2)NC(C)=O)C1 Cc1cc(OCC(=O)NC2CN(C(=O)C(C)OCC3CC3)C2)c(C)c(C)c1 C(C)(CNC(c1cnc(S)[nH]1)=O)(C(C)C)NC(CC1(C=C)CC1)=O Cc1nc(C(=O)NCCN(C(=O)C2=CC(O)CCC2)C(C)C)c2ccccn12 CCC(C(=O)N(CC(O)CNC(=O)CCC1CCCCCC1)C)C(F)(F)F c1(CNC(CN(C(=O)C(C)C2CCC2)CCCC)=O)cn(C)c(=O)nc1O CC(c1ccco1)=CC(=O)NC(C)CNC(c1cnn(C(C)(C)C)c1C)=O C1(ONC(c2n(CC#C)ccc2)=O)CCC(O)C1O.N12CCCC(C1)C(C)(C)C2=O N1(C(c2[nH]cc(C)c(=O)c2C)=O)CCC2CN(C(C3CSCCS3)=O)C2C1 C(C(=O)NCC1CN(C(C2(C(N)=O)CC2)=O)CC1(F)F)(c1ccccc1)=C(C)C C12(C(=O)NC(C(=O)NS(C)(=O)=O)C3CCCC3)CCC(C(=O)NC3CC3)(CC1)C2 N1(C(c2c(C)cc(C(C)C)s2)=O)CCN(C(C2COCCC2(F)F)=O)CC1CO C12(CNC(CNC(C(CC)CC)=O)=O)CCCN(C(c3ccnc(C)c3)=O)C1C2 C1(C)(NC(C2OCCN(C(C(CC)(C)O)=O)C2)=O)CCC(C)=C(C)C1 C(=O)(C1=CCCC1)N(CC(=O)NCCC=C=C)CCOC N1(C(c2n(C)ncc2C2CC2)=O)CC2(CCCN(C(=O)C(O)C(C)(C)C)C2)C1 c1(CC(=O)NCC(CNC(C(CO)N(C)C)=O)CO)ccc(Cl)cc1F C#CCC(C)(C)C(=O)N1CC(O)(CN(C(=O)Cn2nnc(=N)[nH]2)C)C1 C1(NC(c2ccc(C3CC3)o2)=O)CC2(C1)CC(NC(C1CCCSC1)=O)C2 C1(NC(CCN(C(CC)CC)C)=O)CC12CCC(NC(c1ccoc1)=O)CC2 CC(CC(C)N=c1[nH]c(N2CC3SCCC3C2)nc2ccccc12)C(F)(F)F c1(SCC(=O)NC2CC(NC(C3C(C)(C(F)F)C3)=O)C2)ccncc1 C1(C)(CCC(=O)NC(C2CCOCC2)C)CCCN1C(=O)CN1CCCCC1=O C=CCCN=C(NCC(C)(CO)OC(C)C)N1CCCC(OCC)C1 Cc1ccnnc1C(=O)NCc1ccc(CNC(=O)CN2CCCC2C)cc1 N1(C(c2ncn(C)c2)=O)CC2CC1CC2Cc1ccccc1F.C1(=O)CON1 N1(C(C(CC)(F)F)=O)CC2CC(C1)CN(C(=O)CC13CCC(C)(C1)OC3)C2 C=CCCCCCCCC(=O)NCC1CC1NC(c1cc2sc(Cl)cc2[nH]1)=O N1(C(CCC2(NC(c3cc(C)nc(O)n3)=O)CCCC2)=O)CCC(F)(F)C(F)C1 c1(CC)cnn2ccc(C(=O)NC3CCOCC3NC(C3CC(C)(F)C3)=O)nc12 C(=O)(C1CCCc2nccn21)NC(CCC)CNC(c1cncc(C(C)=O)c1)=O C1(C(C(N2CC(O)(CC=C)C2)=O)(C)C)CCCN(C(C2CC3(CC3)C2)=O)C1 c1(N(CC(=O)N(C(C)CCNC(=O)CNC(N)=O)C)C)ccc(Br)cc1 C(=O)(C1=NOC(COC(C)(C)C)C1)NCC(CC)(C)NC(C1(C(C)C)CC1)=O C1(C(=O)NCCC2CCC(NC(CCc3n(C)cnc3)=O)C2)CCC2CC2CC1 C1(OC)(CNC(C2CCC2C)=O)CCN(C(c2cccnc2N(C)C)=O)CC1 CC1CN(C(c2n[nH]cc2-c2ccccc2)=O)CC1NC(=O)Cc1n[nH]c(=N)s1 N1(C(CCOCC#C)=O)CC(C)N(C(=O)CC(C)(C)C)CC1C C1(CNC(c2c(CNC(c3c(C(C)C)ocn3)=O)noc2)=O)CCCCN(C)C1 n1(CC)nc(C(=O)NC(CNC(=O)CC2(CSC)CC2)CO)c(C)n1 c1(OC)ccc(I)c(C(=O)NCC2CC(NC(=O)CNC(C)=O)C2)c1 C1(C2N(C(C(C)N(C)C)=O)CCC2)CCN(C(c2ncn(C)n2)=O)CC1 c1(C(=O)NC(CCCCNC(CCCCC=C)=O)CO)cnc2[nH]nnc2c1 c1(C(=O)NCC(C2CC2)NC(c2ncn(C)c(=O)c2)=O)nc2cc(O)ccc2[nH]1 c1(N2CCCC(C)(NC(=O)CCc3cccs3)C2)nc2ncc(Cl)cc2o1 C1(C(=O)NC2(CC=C)CCC2)CCCCC1(C)NC(c1cccn1CCC)=O C(N=c1cc(NCC(c2ccc(F)cc2)(C)C)nc(C(C)C)[nH]1)c1ncc(C)[nH]1 C#CCCC(C(=O)NC(CN(C)C)CCO)NC(C1C=CCS1)=O c1(CC)cc(C(=O)N(CC)CC2CCCCN2C(=O)CC(C)SC)cc(O)n1 CCC(C)(CC(=O)N1CCN(CC(C)NC(=O)C=C(C)C)CC1)C(=O)OC N1(C(c2c(C)cc(CC)o2)=O)CCN(C(C2Cc3nccn3C2)=O)C2CCCC12 CC(C)(C)C(C(=O)NCC1CCC1CNC(C1C2(CC2)C12CC2)=O)NC(N)=O C1(N(C(C(OC)OC)=O)C)CCC2CN(C(=O)C=C(C)c3ccco3)CC12 CC#CCCCC(=O)N(C)CC1CCN(C(=O)C2=NOC(C3(O)COC3)C2)C1 C(=O)(C(CO)C(C)C)NC(CNC(c1cc(C)c(C)s1)=O)(C)C Cc1ccc2c(c1)SC(C(=O)NC1CCCN(C(C34CCC(CO3)C4)=O)C1)C2 C1(Cl)(C(=O)NCC2N(C(C(CC=C)C)=O)CCC2)C2CCC(=O)C12 c1(NC(C23CN(C(c4c(CC)cccc4)=O)C(C2)C3)=O)cccn2cc(C)nc12 C1(NC(COCC=C)=O)CCCCCC1NC(c1c(C)nsc1NC)=O C1(NC(CCOC)=O)CC2CCC1N(C(C1CCC(CCO)CC1)=O)C2 C(=O)(CC(C)C(=O)N1CC(CC(=O)NCC2(CCO)CC2)CC1(C)C)OCC C1(C(=O)NCC2CCN(C(c3cc(C)nc(C)c3)=O)C2)CCc2ccccc2O1 N1(C(C2C(C)OCC2)=O)CC2COCCC2(NC(=O)CS(C)(=O)=O)C1 c1(C(=O)NC2CCCC(NC(c3ncc(C)cc3F)=O)C2)[nH]nc2ncccc12 c1(N2CC(C)C(O)C(C)C2)nc(=NCCc2ccc(Br)cc2)[nH]c2ccccc12 N1(C(CNC(C)=O)=O)CC(N(C(=O)Cc2cccc(C(N)=O)c2)C)C(F)C1 CC(Cl)(Cl)C(=O)NCCC1CCC(NC(=O)Cn2nnc(=N)[nH]2)C1 C(N=c1[nH]c(=NCC(C(C)C)C(C)C)[nH]c2c1CCCCCC2)c1c(C)ccnc1 C1(NC(=O)C#CC2CC2)CCC2CCN(C(=O)CSc3nc[nH]n3)C1C2 c1(N2CCC3(C)C(C)(C2)C3(F)F)nccc(=NCCCCC#N)[nH]1 CCCCCCCCc1cn(CC2CCCN2C(=O)CC(C)F)nn1 c1(C(=O)NC2C(NC(C(CC#C)O)=O)CC2)ccc(CC)c(N)c1 c1(-n2c(C3CC(OC)C3)nc(-c3ccccc3)n2)ccc2ncsc2c1 CC(C)CCC(C(=O)N1CC2(C=CCO2)C1)NC(=O)CSC(C)(C)C N1(C(CCC2CC(OC)C2)=O)CC2CN(C(=O)C(C(C)(C)C)NC(C)=O)CC2C1 C=CC(CCC)CC(=O)N1CCCCC(CCC(=O)NC(C2CCCCC2)C)C1 C1(NS(C)(=O)=O)CCCC1CNC(=O)Nc1csc(C(N)=O)c1 Cc1cc(N)cnc1C(N1CC(NC(c2ccnc(C3CC3)n2)=O)C2(CC2)C1)=O C(=O)(C1=NOC(C)C1)NCCCCC(C)NC(CC(=C=C)C)=O C1(CNC(CCC)=O)CN(C(=O)Cn2cc(CN(C)C)nn2)CCO1 N1(C(C(C)=CCN(C(c2ccn(CCC)n2)=O)CCO)=O)CCCCCC1 c1(CC)cnc(C)c(NC(=O)C(c2cccs2)NC(C2CNC(=O)N2)=O)c1 S(=O)(=O)(c1ccc(Cl)nc1C)N1CC(F)CC(C(=O)NC(C(=O)OCC)C)C1 C1(NC(C(=O)NC2C(n3c(C)cc(C)n3)CCCC2)=O)CCC2(CCC2)C1 c1(C(=O)NC2CCCN(C(CN(C3CCSC3)C)=O)C2)cccc2cc(O)ncc12 CCCCCCC(c1nnnn1C)NC(N1CCC(C)(NC2CC2)CC1)=O C1(NC(C(C)NC(=O)CCC2CC2(C)C)=O)CCC2CCCC1O2 c1(NC(C2(C(=O)OCC3CC3)CN(C(=O)COC)C2)=O)ccc(C2CCC2)nc1.CC C(=O)(C(F)(F)CC(C)C)N1CC(O)(CCNC(C(C)NC(=O)NC)=O)C1 c1(OC)ncnc(C(N2CC(NC(c3cn(C(C)C)cn3)=O)C(C)(C)C2)=O)c1F N1(C(CCc2nc(C)sc2)=O)CCN(C(C2CC2C)=O)C2CS(=O)(=O)CC12 c1(S)cccc(C(=O)O)c1F.c1(CN(CCC)C(C2CC(N)C2)=O)c[nH]c(=NC)s1 C1(C)(C(N2CC(C)N(C(c3sccc3Cl)=O)CCC2)=O)COc2ccccc2O1 N1(C(c2c(C)nc(CC)o2)=O)CC2CC1CN2C(=O)COCCOCCO N1(C(c2c(CCC)nns2)=O)CCCCC1CNC(c1cc(C(C)(C)C)c[nH]1)=O c1(CCNC2CCCN(C(C(C)N(C)C(C)C)=O)C2)nc2ccccc2s1 C=CCCC(C)(C)C(=O)N1CCC(CC(N2CC(C)(C)C2COC)=O)C1 C1(C(=O)NC2C(NC(=O)CCc3ncc(F)cn3)COC2)CN2CCCN1CC2 C1(NC(Cn2c(C(C)C)ncc2)=O)C2CN(C(c3cscc3Cl)=O)CC12 C1(NC(C2(N(C(CCCC#C)=O)C)CC2)=O)CC(C)N(C)CC1C c1(CC)ccc(CONC(C2CCCN2C(c2ccoc2)=O)=O)cc1 N1(C(c2cccc(CC)c2)=O)Cc2cccn2CC(C(=O)NCCOC(C)=O)C1 c1(C(N(CCNC(C(c2ccccc2)C)=O)CC2CC2)=O)cn(C2CCC2)nn1 CC1CCCN(C(c2cn[nH]c2)=O)C1CNC(=O)Cc1csc(Cl)n1 c1(NCC2CCC(CC)CC2)[nH]c(=NCc2ccc(N)cc2C)nc2scnc12 C1(C(=O)NC2CCC(c3nc[nH]n3)CC2)CC2(CC(NC(c3ccoc3)=O)C2)C1 c1(N(C(CC2N(C(c3ccc(OC)cc3)=O)CCC2)=O)C(C)C)ncc(I)nc1Cl c1(C(N2CC(NC(c3ccc(-c4ccco4)o3)=O)C2)=O)ccc(Cl)[nH]1 C1(CCC(=O)NC(CNC(CSCCCC)=O)CC)CCCCC1 O=C1Cc2c(N3CC4(CCCN4Cc4ccc(I)cc4)C3)ncnc2N1 C1(N(C(Cc2c(C)n(C)cn2)=O)C)CCN(C(c2cnc(O)n2C)=O)CC1C Cc1cnc2c(C(N3CCCC34CN(C(=O)C(O)C(C)(C)C)C4)=O)cnn2c1 CCS(=O)CC(=O)NC(C)(C)CC1CCN(C(C2CC(F)C(=O)N2)=O)CC1 c1(-c2ccc(CC)c(F)c2)ccn2cc(C(=O)NCc3noc(CC)n3)nc2c1 c1(C(=O)NCCC(C(C)C)NC(c2cn(CC)nc2)=O)cccc2c1C(=O)NC2 C(=O)(CCCCNC(=O)C(C)NC(=O)NC)N(CC)CC C1(C(N2CCC(CCNC(C=CCOC)=O)C2)=O)CCN(C2CCSC2)CC1 N1(CCOC)C(=O)NC(c2cc(Br)cc(OC)c2O)C2=C1CC(C)(C)CNC2=O N1(C(C(COC)OC)=O)C(CNC(=O)C(=Cc2cn[nH]c2)C)CC2COCC12 c1(OCC(=O)NCC2C3CCC(C3)N2C(=O)CC2CCC2)ccc(F)cc1F C(CCNC(=O)Cc1cncs1)(C(=O)NC(c1nn[nH]n1)C1CC1)OC C1(CCC)CCC(C(=O)NCC2CCN(C(=O)CCc3nccs3)C2)CC1 N1(C(c2c(C)nco2)=O)C(C(N2CCN(C(=O)N(C)C)CC2)=O)CC2CC12 C(=O)(CCCN=c1nccc[nH]1)N(CC(C)CNC(=O)C(F)(F)c1cscn1)C C1(O)(COC)CCCN(C(c2cnn(C)c2)C(=O)NCCSC)C1 c1(C(N2CC(C(N(C3(C#C)CC3)C)=O)C(C)C2)=O)occ2c1CCC2 C(=O)(CC(C)(C)N(C)C(=O)OCC(C)(C)C)NC1(C)C(SC)CCC1 CC1(C)CCN(C(=O)CCC2CC2(F)F)C1C(=O)NC1(CC2CC2)CC1 c1(CN(c2cnncc2Br)C(c2c(CCC)n[nH]c2)=O)cccc(C(F)(F)F)c1C Cc1csc(=O)n1-c1ccc(CN2CC(OCC3CCCOC3)C2)cc1 C1(CC(=O)N(CCN(C(c2cc(C)ncc2)=O)C)C)CCn2cncc2C1 N1(CCNC(C2(F)CCCCC2)=O)CCN(C(=O)CC2CC2)CC1 CCC(CNC(c1cn(C2CC2)cn1)=O)(CC)NC(c1nnn(C)n1)=O C(CCC(C)C(=O)N1CCN(C(c2ccc(C(N)=O)cc2)=O)CC1CCO)OC c1(C(=O)NCC(N(C)C(c2ccc(F)cc2CO)=O)C2CC2)ccc(C#N)cc1 CN1CCC(NC(c2cnn(C)c2-n2cnnc2)=O)c2ccccc21 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(NC(c2cc(Cl)ccc2C)=O)C(O)C1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCc2ccccc2C(NC(=O)C=CCCC)C1 CCC(Cc1ccccc1)CC(=O)NCCCN(C)C(c1cccnc1F)=O C1(CNC(C2(C)C(C)C2)=O)CCC(N(C(=O)COC2CCCC2)C)CC1 C1(CNC(CC=C)=O)CC2CCC(C1)N2C(=O)C(C(C)C)OC CC1CCc2c(C(=O)NCC(O)CNC(C34CC(C3)C4)=O)csc2C1 C1(C(C)C)N(C(=O)CC2CCC2)CC12CCN(C(C1C3CCC(F)(F)C13)=O)CC2 c1(CNCc2cnc[nH]2)ccc(O)cn1.C12CN(C1)C(=O)C2 N1(CC)CCc2cccc(CCC(=O)Nc3ccc(C(C)(C)C)cc3I)c21 c1(CC(=O)N(C2CCCN(C(C3CC4C=CC3C4)=O)CC2)C)c(C)nn(C)c1C c1(CCC)nc(C)c(C(=O)NCC2CN(C(C3CSCN3C)=O)CC2C)s1 c1(CC)cccc(C(N2CCC(NC(c3ccc(C)c(O)c3)=O)CC2C)=O)c1F C1(OC)CCC2(C(N3CC(C)(NC(=O)COC4CCC(C)CC4)C3)=O)CC12 C1(CNC(C(CC)OCC)=O)CN(C)CCN1C(c1cccc(O)n1)=O N1(C(CCC)=O)CCC(c2cn(C(C)Cc3ccccn3)nn2)(C(=O)OC)C1 C#CC1(C(=O)NCC2(CO)CCCO2)CCN(C(=O)CCCOCCOC)C1 C(=O)(C1(C)CCCc2ccccc21)NCC1N(C(C2C(=C)CC2)=O)CCCC1 n1(CC(=O)NC2(CNC(=O)CC3(n4cccn4)CC3)CC(OC)C2)cnccc1=O c1(C(C)C)cc(C(=O)NC2CCC(CNC(=O)C(C)(C)NS(C)(=O)=O)C2)no1 O=C(C(F)(F)CO)NCC1CCCN(C(C2CCCN(S(=O)(=O)C(F)F)C2)=O)C1 C(CC(=O)NC1CC1NC(=O)C(C)=C1CCCC1)N(CC)CC CCC(CCOC)C(=O)NCC1(C)CCCN(C(=O)COC2(C)CCCC2)C1 C1(C(C#C)C)CCN(C(C2(C(C)NC(=O)C(O)CCSC)CCC2)=O)CC1 C1(c2nnc(N3CCOCC(C)(F)C3)n2CC2CC2)CCCC2CCCCC12 C(C(C)(CC)C(=O)Nc1cccc(C(N)=O)c1)NC(CNC(=O)OC)=O c1(C(=O)NCC2C(CNC(c3c(C)occ3)=O)C2)cc(=O)n(C)cc1Br c1(C(N(CC)Cc2cc(C)nn2C)=O)nc2c(s1)CCCCC2 N1(C(=O)Cn2cnnn2)CCN(C(=O)CN2CC3CC3C2)C2CC12 c1(NCC2CN(C(CNC(CC(C)(C)C)=O)=O)C2)ncc(S(C)(=O)=O)cc1Cl Cc1n[nH]cc1C=CC(=O)NCCCNC(=O)C(C)Cc1ccco1 c1(NC(C(C)OC(C2(C)CCCO2)=O)=O)nc(C2CC2)ncc1Br c1(NCCC2CC(NC(C(CC)OC)=O)C2)ncc(S(C)(=O)=O)cc1Cl C(C(C)(CC)CO)N.CCCCOC(=O)NCCSCC N1(C(C2(NC(c3cc(C)no3)=O)CC(F)(F)C2)=O)CC2CC3CC2C1C3 C1(N(C(c2cnc(O)[nH]2)C2CC2)CC)CCCN(C(=O)CCC2(C)CC2)CC1 CC1=NOC(CC(=O)NC2CC(OCC(=O)NC(C3CCCC3)CO)C2)C1 C1(CNC(C(CC=C)CC=C)=O)CN(C(=O)Cn2cnnc2)C2CCCCC12 c1(CC)ccc(CCC(N2C(CNC(C3(C)CCC(=O)N3)=O)CC3CC23)=O)cc1 C1(NC(c2c(OC)cnnc2)=O)CN(C(=O)COc2cccnc2)C(C)(CO)C1 c1(C(=O)NCCNC(c2cc(C)n(-c3ccn(C)n3)c2C)=O)cc(F)c(N)cc1F N1(C(=O)C(F)(F)CN2CCCC2)CCCCCC(NS(=O)(=O)c2ccc(Cl)cc2)C1 c1(OC(C)C)cccc(C(=O)NCCCCN(C)C(c2ccc(C(N)=O)s2)=O)n1 C1(NC(c2ccc(Cl)c(OC(F)F)c2)=O)CCN(CCc2ccccc2)C(=O)C1 N1(C(C2C(C=C)C2)=O)CCC2(CCC(NC(=O)COc3ccc(F)nc3)CC2)C1 C1(NC(C(Br)=C(C)C)=O)CCCCC12CCCN(C(C1CCC1(C)C)=O)C2 C12(NC(C(C)OCCOCC)=O)CCOC(NC(C3(C)COC3)=O)(C1)C2 c1(C(C)C)nc(=NC2CC(C)N(C(C3CN4CCCN3CC4)=O)C2)s[nH]1 C1(C(C)C)CN(C(=O)CC(C)(F)F)CCN1C(=O)CC1CC1 c1(CCC(=O)NC2(C)CN(C(C3CN(S(CC)(=O)=O)C3)=O)C2)c(C)noc1Cl CCCCCC(C)CC(=O)NC1CN(C(=O)CCc2nc(=N)[nH][nH]2)CCC1CO CCCCCC(=O)NC1CC(CO)N(C(=O)CC2(N(C)C)CCC2)C1 C1(NC(C2(C)CC2(F)F)=O)CCC2CN(C(=O)CCc3ccc(O)nc3)CC2C1 C1(C(N2CC(C)(C)C(NC(C3CC(F)(CO)C3)=O)C2)=O)CCc2ncncc2C1 c1(C(=O)OCc2ccc(Cl)s2)ccc(F)c2cccnc12 C12(C(N3CCC(CC(=O)NCC(F)C4CCC4)CC3)=O)CCC(CC1)CO2 C(CC(=O)NCC(C)N=[N+]=[N-])(CC(C)C)NC(c1ccc(C=C)cc1)=O n1(CC(=O)NCC2CN(C(C(C)C3CCCO3)=O)C2)cc(CO)nn1 C1(N2CCCC2)(CN(C)C(=O)NCC2CC(F)C2)CCOCC1 c1(C(=O)NCCCCNC(C2(CC(C)C)CCC2)=O)cn(C)nc1C(C)C N1(C(C(C)SC)=O)CCCC12CCN(CCNc1nccc(C)c1[N+](=O)[O-])C2 CON(CCC(=O)NC(C)CN(C)C1CC1)C(=O)C(C)CC1CC1 c1(CC)ccc(-c2nc(-c3cccnc3)nn2-c2ccc(C(C)(C)C)cc2)cc1 C=CCCC(C(=O)OC)NC(C1CC(C)(C)CN1C(=O)C(CC)SC)=O CC1CCN(C(C2CSCN2C(=O)C2CC2)=O)CCN1C(c1ccncc1F)=O Cc1c(F)ccc(C(=O)NCC(C)CNC(C23CCOCC2C3)=O)c1N CCCC(C(=O)NCCN(C(C1CCC1(F)F)=O)CC)c1ccccc1 CC(Cc1cccc(Cl)c1)CC(=O)NC1(CNC(=O)C(C2CC2)N(C)C)CCC1 C(=O)(C1=CCC(NC(c2cc(F)ccc2F)=O)C1)N(C)CC1CCC(F)(F)C1 c1(SC)cc(C)ccc1C(=O)NCCNC(C1(C)CC(=O)C1)=O N1(CC(=O)NCC(CC)NC(c2scnc2COC)=O)CCN(C)CC1 C(=O)(CCC(O)C(C)(C)C)N(C1CN(C(CCc2cccc(OC)c2F)=O)C1)C c1(N(CC(c2ccc(Br)cc2)C)C)nc(=N)[nH]c(=NC(CSC)c2ccccc2)[nH]1 C(C)(C)(C(=O)NC(C)C(=O)NCC(O)Cn1cccn1)OC(C)C Cn1cc2c(n1)CCCC2C(=O)NCCOCCCNC(=O)CCC1CCCO1 Cn1nc(-c2ccccc2)cc1C(=O)NC1CC(NC(C2C=CCS2)=O)C1 N1(C(C)=O)CCN(C(C2CCCCO2)=O)CC1n1cc(-c2sccc2CO)nn1 CON(CCC(=O)N(C1CCNC(=O)CC1)C)C(=O)c1c[nH]cc1C C1(CC(C)O)CCCCN1C(C1CN(C(=O)COc2ccccc2)CC1C)=O N1(C(C2(C#C)CCN(C(=O)CP(C)(C)=O)C2)=O)CCC(F)(F)CC1C C1(CNC(c2cccc(Cl)c2C(F)(F)F)=O)CCN(C(c2cocn2)=O)C12CC2 c1(C(=O)NC(CC)CNC(c2cc(C)sn2)=O)ccc(=O)n2c1COCC2 N1(N(C(C)(C)C)C)CCC2(CCCC2C=O)C1.C1(C2CC2)(COC=O)CC1 N1(C(C(=O)NC2CCC(C(=O)OC)C2)c2nccs2)CCC(C2CC2(F)F)CC1 c1(OCC(=O)NC2CCCNCC2)cccc(SC(F)(F)F)c1Cl C1(NC(=O)CCn2cc(CO)nn2)CC2(C1)CC2NC(C1CCCC(=O)N1)=O C=CC(CC)CC(=O)NC1CCCN(C(=O)COc2ccc(Cl)c(C)c2)C1 C12(NC(CC3CC(OC)C3)=O)CCC(CN(C(=O)C(C)=C3CC3)C1)C2 C1(CSC)CN(C(=O)CCn2cnc(=N)[nH]2)CCN1C(=O)OC(C)(C)C c1(C(=O)NC2CC(O)(CNC(C3(C)CCCCO3)=O)C2)cccc(N)c1Br CC1CN(C(=O)C=Cc2cc[nH]n2)CCCN1C(C1CC2CCC2C1)=O C1(NC(C2CCCN(C(N)=O)C2)=O)Cc2ccccc2C1NC(=O)CC1CC1 Cc1nc(F)ccc1CN1CCC2(CC2C(=O)NC2CCC(=O)NC2=O)C1 N1(CC(=O)N(C)CC2CCN(C(C3(C4CC4)CC3)=O)C2)CC2CCC1C2 C(=O)(C(O)C1=CCCCC1)N(C1CCC(NC(=O)C(C)(C)CCSC)CC1)CC C1(NC(=O)C(O)c2cnc[nH]2)COCC1n1cc(-c2cnn(CCF)c2)nn1 c1(C(=O)NCCN2CCCN(C(=O)C(O)CF)CC2)ccnc2ccccc12 C=CC(CC)CC(=O)NCC1(CNC(c2scnc2C)=O)CCC1 C1(NC(Cn2cc(C(=O)NC)nn2)=O)COCCN(c2nnc(C(F)(F)F)s2)C1 N1(C(CCCOC(C)(C)C)=O)CCSC(C(=O)NCc2cscn2)C1 Cc1cc(C(N2CCCCC2CN(C)Cc2noc(C)n2)=O)c(C)c(C)c1 CC1CN2CCN1C(C(N1CCC(NC(=O)CN3CCCCC3=O)C1)=O)C2 C1(NC(C2(SC)CCC2)=O)C(C)CN(C(C2CCc3nn[nH]c3C2)=O)CC1C CCCCC(CCC)N=c1[nH]c(=NCCC(=O)NC)[nH]c2c1CC(C)CC2 C1(C(N(C)Cc2cc(C)no2)=O)CCN(C(C2CCC2(F)F)=O)C(C)C1 c1(CN(C(C)(C)C(=O)O)CCCC)cc(C2CC2)on1 c1(CNC(C(=O)N(C2CCNCC2)CCC)=O)nc(OC)cc(OC)n1 N1(C(CNC(CNC(c2ccc(C(C)C)o2)=O)=O)=O)CCCC1(C)C(C)O c1(OC)ccc(C(N2CC(NC(=O)Cn3ncnn3)C(C)(C)C2)=O)c(N)c1F N1(C(c2ccc(=N)[nH]c2Cl)=O)CCCC(NC(c2ncc(Cl)cc2F)=O)C(F)C1 C1(CCC)(NC(c2coc3c2COC3)=O)CCN(C(=O)Cc2nc(C)cs2)CC1 C(C1CCc2ccccc21)NC(c1n(CCC)nnn1)c1cc(CO)on1 C1(C(N(CCN(C)C(C2CC2C(N)=O)=O)C)=O)C2CN(CC(F)(F)F)CC12 C=C(Cl)CC(C(=O)NCCC1C=CCC1)NC(=O)CC12CCCC1C2 N1(C(c2n(CC)ccc2)=O)CC2(CCCC2NC(c2cn[nH]c2)=O)C1 C(=O)(C(=O)NOC)NC(CNC(C1(C(CC)=O)CC1)=O)CC C(=O)(C1=COCCC1)NCC1C(CC)CCN1C(=O)CC(F)(F)c1ccccc1 c1(NC)cncc(C(N2CC(CNC(c3cc(SC)oc3C)=O)C(C)C2)=O)c1 CC(C)CCC(O)C(=O)NCC1(CNC(=O)C(C2(O)CCCC2)F)CCCCC1 CCCC(CC(C)C)C(=O)NCc1cccc(CNC(C2CNC(=O)N2)=O)c1 C1(NC(CC(C)OC)=O)COC2CN(C(c3ccc(SC)cc3Cl)=O)CC12 CC1(C)CC(=O)NCC1C(=O)NC1C2CC1CN(C(=O)COc1ccon1)C2 C1(O)(C(N2CC(C(C)NC(C34CC(CO3)C4)=O)C2)=O)CC2CCC1C2 c1(C(=O)NC2CN(Cc3cccc(OC)n3)CC2O)ccc(Cl)nc1Cl c1(OCC)cc(C(N2CC(C)C2)=O)ccc1NC(=O)C(C)OCCN(C)C.CC.ON C1(NCc2n(C)cnn2)C(NC(C2CCN(S(C)(=O)=O)CC2)=O)CCC12CCC2 C1(NC(C2(C)CC(NC(C3CC(OC)C3)=O)C2)=O)CC2CC1OC(=O)N2 c1(C(N(CCNC(C2N(C(C(C)C)=O)CCCC2)=O)C)=O)cc2c([nH]1)CCOC2 C=CC(C)(O)C(=O)NCCC(C(C)C)NC(c1ccn(C(C)(C)C)n1)=O C(CC(=O)NC1CCCN(C(c2cnc3c[nH]nc3c2)=O)C1)(C(F)(F)F)OC C(=O)(CCC1CC1)NCCN(CC(C)O)C(C1CCN1C1CCCC1)=O.C(C)(C)C N1(C(c2nccc(C)n2)=O)CCC2(CC1)CC2CNC(C1CCC(C(N)=O)C1)=O C1(CCN(C(=O)CC(C)(C)O)C)CCCCN1C(=O)CC1CCCOCC1 c1(N(CCNC(=O)OC)C)ccccc1C C1(C(=O)NCC2CCCC(C)O2)CN(C(c2cc[nH]c(=N)n2)=O)CC1(F)F N#CC1CN(Cc2cc(Cl)cc(Cl)c2O)CCN1C(c1ccc(O)c(Cl)c1)=O c1(C(=O)NCC(C)(C)N(C)C)ccc2c(c1)nc(O)n2C1CCCC1 C1(CNC(c2nc(C)nn2C)=O)CC2OCCC2N1C(c1ccc(C)c(F)c1)=O C1(C(N2CC(C(=O)OC)C2)=O)C(O)CCN1C(c1csnc1C)=O Cc1ncnc(O)c1C(=O)NC12CC1CN(C(=O)C(c1cnccn1)C)C2 c1(C(=O)NC2CN(C(c3ncn(C(C)C)n3)=O)CC2C)cccc(F)c1C#N CN1CC2CCCC(C1)N2C(C1C(O)CCN1C(=O)CCC(C)(C)C#N)=O Cc1nc2ncccc2cc1C(N1CCC2(CC1)CN(C(C1CCC1C)=O)C2)=O c1(C(=O)NC(CC=C)CNC(c2cc(CO)[nH]n2)=O)cccc2nc(CO)[nH]c12 Cc1ccc(C(F)F)cc1C(=O)N(C)CCNC(=O)C(=O)C(C)C c1(C(=O)NCC2(F)CC(NC(C(C)O)=O)C2)ccc(S(C)(=O)=O)s1 N1(C(C(C2=CCCC2C)NC(=O)CCCn2ccnc2)=O)CCC(C)OC(C)C1 C#Cc1cc(Br)cc(Cl)c1NC(=O)CC(c1ccccc1Cl)Nc1ccccc1 C=CCC(CNC(c1coc(C)n1)=O)NC(c1cc(-c2csc(CO)n2)c[nH]1)=O N1(C(CNC(C(C)(C)C)=O)=O)CCCC2(CCCN2C(=O)C=Cc2cc[nH]n2)C1 Cn1cnc(S(=O)(=O)NCCC(=O)NCC2CC2NC(=O)CCCCCN=[N+]=[N-])c1 CCCC(C(O)C(=O)NCc1nccn1C(C)C)NC(=O)C(C1(C)CC1)SC c1(C(=O)NCC2CN(C(c3cc(Br)ccn3)=O)C2)nccn2c(Br)cnc12 CC1CN(C(c2cn(CCO)nn2)=O)CCC1NC(C12CCOC(C)(C1)C2)=O Cc1cccc2nc(CCNC(=O)Nc3noc4c3CCC4)cn12 c1(CC(=O)NC2CCC(N(C)C(C3CCCC3)=O)C2)ccc2c(c1)CCCS2 S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NC1N(C(C(C(C)C)F)=O)CCC1 CCC(C)CC(C(=O)N1CCC2CCCC12)NC(=O)CCCOC(C)=O CC1(C)C(CC(N2CC3(CCC3)C2)=O)CCN1C(c1ccc(CC#N)cc1)=O Cc1csc(CN(C)C(c2sccc2CNC(c2cnc(O)o2)=O)=O)n1 N1(C(C)=O)CCN(C(C2CCC(=NO)CC2C)=O)C(CCO)C1 c1(OC2CCSC2)ccc(C(=O)Oc2ccc(C(C)C)cc2)cc1 CS(=O)c1cccc(C(=O)NCC2CCCCN2C(=O)C2=CCCC2)c1 c1(C(=O)NCCN(C(C(CC=C)F)=O)CC(C)O)cccc2c1nc(O)n2C CCCC(C)CC(=O)NC1CCCC(NC(c2ccccc2-n2cnnn2)=O)C1 C1(CC=C)(NC(=O)CNc2nccs2)CCCN(C(C2CCN(C)C2)=O)C1 c1(NC(CNC(C(C2CCOC2)OCC)=O)C(C)C)ncc(F)cn1 Cc1oc(CO)cc1C(=O)N(C1CCC(NCc2ncnn2C(C)C)C1)C C(N=c1cc(C)nc(NC2CC3CC3C2)[nH]1)c1c(CC)nco1 N1(C(C2C(C=C(C)C)C2(C)C)=O)CC2(CC2)CC1CNC(=O)C(C)O CCC(CC)(CC)C(=O)N1CC2CCC(CNC(=O)CC3(C)CCOC3)C2C1 CCC(C)CC(=O)N1CCN(c2ccccc2O)CC1.C1C(=O)N1C1CC1 c1(C(=O)NCC(C)NC(C2(COC)COC2)=O)ccn2cc(C3CC3)nc2c1 N1(C(=O)Cc2ncccn2)CCCCC2(CCN(C(=O)C(O)C3CCCC3)C2)C1 C#Cc1cccc(C(=O)NC2CC3C(NC(C4CCCCC4C)=O)C3C2)c1 Cc1c[nH]c(COC(C)C)c(C)c1=O.C12CCCC1C(C)(C)CO2 C(CCCCCC(=O)N1CC(OCC(C)C)C1)NC(C(C1CCC1)OC)=O CC1CC(CCC(=O)NCC2(NCC3CCC3C(N3CCC3)=O)CC2)C1 C(=O)(CCC(C)(C)C)NC(C(=O)NCCN1CCCC(C)C1)CCF c1(-n2cc(CCC(=O)NC(C)C(C)(O)c3ccccc3)nn2)cc(F)ccc1Br N1(C(CC=C=C)=O)CC(NC(c2ccc(O)cc2)=O)C2(CCOCC2)C1 C1(c2cn(CC(N3CC(C)(C)OCC3)=O)nn2)CCC2CCCCC2C1 Cc1ccc(COC(C)C(=O)NC2CCCC2NC(=O)C(=O)NCCCF)cc1 C1(C(=O)NC(COCC)C)(NC(c2nc(O)sc2C)=O)CCN(C)C1 Cc1ncc(Cl)c(C(=O)NC2(C)CCN(CCOC(F)(F)C(F)(F)F)C2)n1 C1(NC(c2cc(COC)cn2C)=O)CCN(C(C2COCCC2C)=O)C(C)C1 C(=O)(CS(=O)CCC(F)(F)F)NCCN(C(C(C(C)(C)C)(C)O)=O)C1CC1 C1(CC(N2CC3CC3(CO)C2)=O)CC2C=CC1C2.C123CC(C1)(C2)NC3=O C(=O)(C(F)C(F)(F)F)N(CCCNC(c1cc(C(C)C)[nH]n1)=O)CCO C(=O)(CC(C)C(C)(C)C)N1C(CC(=O)NCCOCC=C)CC(C)(C)C1 O=S(=O)(c1ccc(F)cc1F)N1CC2CC1CN2Cc1ncccc1C(F)(F)F N1(C(c2cc(C)no2)=O)CCC(C)(C)C(NC(=O)CN(C)S(N)(=O)=O)C1 N1(C(C2(C=C)CC2)=O)CCOC2(CCN(C(C3CC3C#N)=O)C2)C1 C(=O)(C(C(C)C)OCC(C)C)NCCCCCNC(C1(CCOC)CCCC1)=O C1(NC(C(C)NC=O)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)CC1F N1(C(C(C)n2cncn2)=O)CC2(CNC(C3(C(C)(F)F)CC3)=O)CC1CO2 C(=O)(CCC(C)(C)C)OCCCNCC1CN(c2cccc(OC)c2)C(=O)C1 C(=O)(C1CCC(N)c2ccccc21)N1CC2C(CN(C)CC)C2C1 CCC(F)(F)C(=O)NCC(c1ccc(OC)cc1)NC(c1conc1C)=O c1(C(=O)NC2C(NC(C(C3CCOCC3)OCC)=O)CC2)cc(N)cc(F)c1 c1(OCCC)ccccc1OCc1nnnn1CCC.C12CCCCC1NC2=O c1(NC2(NC(N3C(c4scc(C(=O)OCC)n4)CCC3)=O)CC2)cncc(O)c1 C(=O)(C(C)CC(=O)N1CCOCC1CN(C(=O)C(=Cc1ccccc1)C)C)OC C#CC1COCCN1CC1CC(OC(C)C)CN1Cc1ccccc1 C1(CSC)CN(C(=O)CCCN(C)C(C)C)CCN1C(=O)CC1C(C)(C)C1(C)C CC(C)(CCNC(=O)Cc1cnc(Cl)s1)NC(c1ccc(C2CCCCC2)o1)=O C1(C(=O)NC(C2CCN(C(C3(F)CCC3)=O)CC2)(C)C)CC2(CCCC2)CO1 c1(CCNC(=O)NC(c2c(Br)ccc(OC)c2)C)nnc2n1CCN(C)C2=O CCC(C)C(O)C(=O)NCC1(O)CC(NC(=O)CC23CCCC2C3)C1 CCCCCCCCC(=O)N1CCC(NC(=O)C=CCN2CCCC2)C(O)C1 Cc1nn(C(C)C)c(NC2CC(C)N(C(=O)Cn3nnnc3C)C2)c1[N+](=O)[O-] c1(C(N(C)CC2CCN(C(C(CC)NC(N)=O)=O)C2)=O)cc(C)n(CC)n1 n1(CC)nc2c(c1C(N1CC3CC1C3NC(=O)CC1CC1C)=O)CCCC2 Cc1cc(=O)ccn1CC(N1CCC(NC(c2snnc2C(C)C)=O)CC1C)=O CC1(C)CN(C(=O)Cn2ccc([N+](=O)[O-])n2)CC1NC(c1nsnc1O)=O C1(C)(C(N2CCCC(C)(NC(C(C3CC3)SC)=O)C2)=O)CCC(C)(C)CC1 c1(CC)cc(NCCC2CCCN(C(c3sccc3Cl)=O)C2)nc(C)n1 c1(C(=O)NCC2COCCN(C(c3c(C)coc3C)=O)C2)cc2ccccc2[nH]1 N1(C(C23C(C)OC(C)(C2)C3)=O)CCC(NC(=O)CSC(F)F)C(C)(C)C1 C1(C(=O)NC2CN(C(C(c3ccc(C#N)cc3)(C)C)=O)C2)CCc2nncn2C1 N1(C(C(N2CC(C)C2)C)=O)CCCCC1CNC(c1cccnc1C(F)F)=O CC(CC(F)(F)F)C(=O)NC1CC2CC(C1)N(C(c1ccccc1C(N)=O)=O)C2 Cc1ccc(C(=O)NCC2CN(C(=O)CCCc3ccccc3C)C3CC23)cn1 Cc1cccc(C=CC(N2CCCC2C(=O)NC2CC(C)N(C)CC2C)=O)c1 C1(C(=O)NCC(C(C)C)NC(c2ccc(CC)s2)=O)Cc2ccccc2C1 C1(CNC(Cc2nnc(C)o2)=O)CC2CCC(C1)N2C(=O)Cc1ccnc(F)c1 c1(C(C(=O)NCCCSC)N(C(C(=O)OC)C)C)cc(-c2ccc(C)s2)[nH]n1 C(=O)(C(O)CC(C)(C)C)N1CCC(OC2CN(C(C(C(=C)C)(C)O)=O)C2)CC1 C1(CN(C(=O)CN2CCC(O)CC2)C)CN(C(c2ccccc2CO)=O)CCO1 CCCCC(CC(=O)N1CCCC1(C)C1CCC1)NC(c1nocc1C)=O C=CC1CC(c2nnnn2C(C)CC)(NCc2ncc(C(=O)OCC)s2)C1 C12CN(CC1C)C(=O)CONC(=O)C2.C(CC(C)(C)N(C)C)=C(C)C c1(OCC(=O)NCC2CC2CNC(=O)CC2CC2(Cl)Cl)ccc2c(c1)CCC2=O c1(C(NNC(c2ccc(C)cc2C)=O)=O)cc(Cl)c(Cl)c(Cl)c1O C(C(F)(F)CC1CC1)NC(C(n1cc(C(C)NC2CCOCC2)nn1)C)=O Cc1nn(CCC(=O)N(C)CCNC(=O)C(c2ccccc2)C)c(C)c1C c1(N(C2CCN(C(C(CCC)OC)=O)C2)C)ncnc2c1cnn2C c1(CCC(=O)NCC(CNC(c2c(C)ncs2)=O)F)c(C)nc2ncnn2c1C N1(C(COCCCCC)=O)CC(CNC(=O)CC2CSC2)(COC)C1 C1(C2C(C)C2)CSC(CC(N2CC(C(O)C(=O)Nc3ccc(C(N)=O)o3)C2)=O)C1 C1(C)(C(N2C(CC)CCC(C)C2)C(=O)NCSc2ccccc2)CCC(C)(C)CC1 C(=O)(C(C)CC(F)F)Nc1ccc(CNC(C=CC(=O)OCC)=O)o1 C1(CC)C(C(=O)NCCC(O)C(C)C)CCCN1C(=O)COC(C)C c1(C(c2nnnn2Cc2cccc(F)c2)NCCCC=C)c(Cl)cc(Cl)cc1Cl N1(C(Cn2ccc(C)n2)=O)CC2CCC(C1)C2CNC(c1cc[nH]c1C)=O CCC(CC(=O)NC(C)(C)CNC(c1n[nH]c(C)c1C)=O)OC CC1(CC(=O)NC2CC3(CCC3)C2)CCN(C(C23CCCCC2C3)=O)CC1 CN1CC(=O)N(CC(=O)NCC2CC(O)CN2C(=O)C(CO)N(C)C)C1=O CC1CN(C(C2(C#N)CCCOC2)=O)CCN1C(=O)Cn1cc(C2CC2)cn1 C1(CC)CC(C)(C)CN1C(c1ccc(Cn2cc(-c3ccncc3)nn2)cc1)=O c1(OC)cc(F)c(F)cc1C(=O)NC(C)CN(C)C(C1CCCC(=O)N1)=O C(CCCCCC(=O)NC)N.C1(CNC(CC(=O)C(C(C)C)=O)=O)CCC(=O)NC1C C1(NC(CCN(CC)CC)=O)CN(C(=O)C(=Cc2cnn(C)c2)C)CC1OC N1(C(C(CC)CC2CCCC2)=O)CC2CCCN(C(=O)C=Cc3cccn3C)C2C1 C(=O)(C1c2ccccc2C2CC1C2)NCC1C(C)(C)CN(C(C2CC2(Cl)Cl)=O)C1 c1(C(=O)NCCCCC2CCCC2)ccncn1.C12CC1C(=O)NC2 c1(C(N(CC(=O)NC(c2ccnn2C)COC)C)=O)ccn(CCF)n1 C1(NC(CCC)=O)CCC2(CCN(C(C3(C4CC4)CC3)=O)CC2)C1 C1(C(=O)N)(CSCC)CCOCC1.C12CN(C1)C(=O)COC2.C1(C)CC1 C1(OC)CC2(C(=O)N(C)CCOCCN(C(=O)CNC=O)C)CC12 Cc1ccc2[nH]cc(NC(=O)C(CC=O)SC(F)F)c2c1.C(C)(C)(C)O C(=O)(CC(C(F)(F)F)NC(=O)CCn1cccc1)NCCC(CC)CO Cn1ccc2sc(C(=O)NC3CC4(CCC(NC(C5CCCS5)=O)CC4)C3)cc12 C(=O)(CCC(CC)OC)NCCn1ccc(C(=O)NCC(CCCC)O)c1 N1(C(Cc2nc(NC(c3cccc(C#N)c3)=O)sc2)=O)Cc2ccc(O)cc2C1 c1(NC(=O)NCC2CCOCO2)cccc(N2CCNC2=O)c1 c1(OC)cc(C=CC(N2CCC(NC(C3C(C)C3C)=O)C(C)C2)=O)ccc1N N(C(=NCCCF)NCC1(C)CCCO1)CC(C)Oc1cccc(F)c1 c1(C(=O)OC)cccc(NC(=O)COC(=O)CC2CNC(=O)C2)c1F C1(C)(CNC(C(C)(F)F)=O)CN(C2CCN(C(C34CCCCC3C4)=O)CC2)C1=O N1(C(C(C)CBr)=O)CCCC2(CCCN2C(=O)C(O)CCl)CC1 C1(C(N2CC(C(C)NC(Cc3c(C)cco3)=O)OCC2)=O)CN2CCCN1CC2 c1(C(=O)NC2CN(C(CSCC(C)=O)=O)C(C)C2)ccc2scnc2c1 C(=O)(C(C)C(F)(F)C(F)F)Nc1conc1CC1(NC(=O)OC(C)(C)C)CC1 Cc1cc(=O)oc(C)c1C(=O)NC1CN(C(c2ccccc2)=O)CCC1CO Cc1cccn2ncc(C(=O)NCC3CCCCC3NC(C3CC4(CC4)C3)=O)c12 C(=O)(CC(C)C(C)(C)C)NCC(C)CNC(c1cccc(N2CCCC2=O)c1)=O Cn1ccnc1CCC(=O)NCC1(CNC(=O)COC2(C)CCC2)CC1 c1(C(=O)NC(CC=C)CNC(=O)C=CSC)cnn2cccnc12 CC(C)CC(C(=O)NC(C1CN(C(=O)C(F)Cc2ccccc2)C1)C)C(C)C Cc1nc(C(=O)NC(C2CCCC2)CNC(=O)C=CC(F)(F)F)co1 N1(Cc2cc(C(=O)OC)nn2C)CC(C)(C)CC1C(=O)NC1CCCCC1OC N1(C(=O)CSc2cccs2)CCCC2(C1)CN(C(C1CC3(CCCC3)C1)=O)C2 c1(C(N2CC(NC(c3ncn(CC)c3)=O)(CO)C2)=O)ccc2cnoc2c1 CC1CCN(CC(=O)NC2CC2CNC(=O)C(C)Cc2ccnn2C)CC1 C1(n2cc(CN(C(=O)Cc3cc[nH]c3)C3CC3)nn2)CON(C(=O)C2CC2(Cl)Cl)C1 CC1(C)CCCC(C)(NC(=O)C2=CC(O)C(NC(=O)C(F)C(C)(F)F)C2)C1 c1(SCC(=O)NCCN(C(=O)C(F)CCCC)CCOC)nnc2ccccn12 c1(CC(N2CCN(C(CC=C=C)=O)CC2CO)=O)c(C)nc(C)nc1O N1(C(c2on(C)c(=O)c2)=O)CCC(NC(=O)CCc2cc(F)cc(F)c2)C12CC2 C1(C(=O)NCC)CCCN1C(=O)CN(C(=O)CC(C)N(C)C)C1CC1 N1(C(CC2CC(OCC)C2)=O)CCC2(CC1)CC2NC(c1cc(C)c(C)[nH]1)=O c1(NC(C2C(F)(F)C23CCC3)=O)cnc2c(c1)nnn2O N1(C(C2CCC(F)(F)C2)=O)CCC2CCC(C1)N2C(=O)C(c1cccc(Cl)c1)O C(=O)(C1=C(Cl)CCC(C)C1)N1CC(N(C(Cc2c(F)ccc(C)c2)=O)C)C(O)C1 Cc1cnccc1CNC(C1CCN(C)CC1)c1nnnn1CC(F)F c1(CN2CC(NC(c3cc(OC)ncc3)=O)C(F)C2)cc(Cl)ccc1Cl c1(C(=O)NCCC(C)NC(c2c(C)nc(O)s2)=O)cc(N)nc(Br)c1 C12(CC)CCCN1N1C(CCC1)CNC2=O.c1(C=O)cn(C)[nH]c1=N c1(C(N(C)CCOCCN(C)C(C2CCS(=O)(=O)N2)=O)=O)coc(S(N)(=O)=O)c1 C1(C(=O)NC(CC(C)C)CNC(=O)Cc2cnn(C)c2)CCOCC12CCC2 C(CS(=O)(=O)CC)NC(CCN(CC#C)C(c1cc(C2CC2)on1)=O)=O C1(CCNC(N2CC(C(C)(C)C#N)C2)=O)CCCSC1 c1(C(=O)NCC2CC(F)(CNC(c3cccnn3)=O)C2)cccc(C2COC2)c1 CC(C)C(CC(=O)N1CCN(C)CC1CNC(c1cc2c(s1)CCC2)=O)C(C)C C12(CNC(C3N(CC)CCC3)=O)CC(CN1C(=O)CCC1CCCOC1)C2 N1(C(C2CCN(C)C(=O)C2)=O)C2CCC1CC(F)(CNC(C1(O)CC1)=O)C2 c1(C(N2CC(C(C)NC(C(C(C)C)C)=O)C2)=O)ccc2nc(O)n(C(C)C)c2c1 C=C(C)CC(C(=O)N1CC(C(=O)NC2(c3cc[nH]n3)CC2)CC1(C)C)NC(C)=O c1(C(N2CCC(NC(CC(COC)C)=O)C(F)C2)=O)cc(C)c2c(c1)CCCN2 c1(CCC(=O)NC(C)CNC(=O)C(c2ccccc2)C2CC2)ccc(Br)nc1 N1(C(C(CC=C)C)=O)CCN(C(C2CC3(C2)CC(C#N)C3)=O)CC(O)C1 CCC(CC(F)(F)F)C(=O)NCC1CC(NC(=O)Cn2cc(C(=O)NC)nn2)C1 C1(C(N(CCCCC=C)C)=O)CCC(C)N1C(c1ccnc(CO)c1)=O N1(C(CCCOC(C)=O)=O)CCN(C(c2c(CO)cnn2C)=O)CC1c1ncc[nH]1 c1(CC)nn(C)c(Cl)c1C(=O)NC1CCCN(C(=O)C(O)CC(F)F)C1 C1(NC(CC2(CSC)CC2)=O)CCCCC1CCC(=O)NC1CCCC1C C(=O)(C1CCc2ccc(Cl)nc21)NC1CN(C(c2scc(S(C)(=O)=O)c2)=O)C1 N1(C(C(CC)OC)=O)CCC(C2(O)CCN(C(C34CC(F)(C3)C4)=O)C2)CC1 C(C(C(C)(C)C)NC(C1(C)CC1(Cl)Cl)=O)NC(Cn1cc(C(=O)OCC)nn1)=O C1(C(N2CC(C(C)NC(c3cc(C4CC4)nn3C)=O)C2)=O)CC(=O)C12CCC2 c1(C(=O)NC2C(CNC(c3n(C)nnc3)=O)C2)c(F)cncc1Cl N1(C(C(F)=CCC)=O)CCOCCC1C(=O)NCCCc1cc[nH]n1 n1(CC)c(N(CCC2CC2)C2CC2)nnc1C(C)CF C1(CN(C(=O)NC(c2ccc(COC)cc2)C#N)C)CCC(CC)CC1 N1(C(COC(C)(C)C)=O)CC2CCC2(NC(c2cc(Br)ccc2OC(F)F)=O)C1 c1(C(N(C2CN(C(CCC=C)=O)C2)C)=O)sc2ccccc2c1Br CCCN(OC)C(=O)CC(C(F)F)NC(c1cc(CC)sn1)=O CN1CC(N(C)C(c2occc2CNC(=O)CCCN=[N+]=[N-])=O)CCC1=O C1(C(N(CCC(C)NC(c2cc(S(C)(=O)=O)c[nH]2)=O)C)=O)Cc2ccccc2O1 C(C(CC(C)C)NC(=O)CN(C)C(=O)C1CC1)NC(Cc1ncc(COC)[nH]1)=O c1(CC(N2CCCN(C(=O)CCn3ccnn3)CC2)=O)ccc2c(c1)CCO2 C(=O)(C(C)CNC(=O)CC1OCCO1)NCC1CN(C(C)=O)C1 C1(NC(C2(C)CC2)=O)COC2(CNC(c3cc(N)ccc3F)=O)CC1C2 Cc1ccc(C#N)cc1C(=O)NCC1CN(C(=O)C=Cc2cocn2)C1 c1(OC)ncc(C(N2CCCC2C(=O)Nc2ccc(I)c(C)c2)=O)cc1Br N1(C(c2c(C)nns2)=O)CC(NC(=O)Cc2ccc(Cl)nc2)CC12CCC2 C(=O)(C(F)C(C)(C)O)N1CCC(CC(=O)NC2C(CC=C)COC2)CC1 CCCCCCCC(=O)NC1CCCC1CNC(=O)Cc1cc2ccccc2o1 C1(CNC(=O)C2=CCC2)CC2(CCN(C(C3CCC4(CCC4)CO3)=O)CC2)C1 C1(C#N)(C2C(NC(=O)NC(CCC)c3ccco3)CCC2)CCCO1 CC(C)(C(=O)NC1CCN(C(=O)C2CC2)C1)c1ccc(-c2cn[nH]c2)s1 c1(C(=O)NCC2(CCC=C)CN(C(C3CCC(C)S3)=O)C2)nc(C)c(C)[nH]1 N1(C(CC2CCCC(C)O2)=O)CC2CC(C)N(C(=O)CC(F)(F)C(F)(F)F)C2C1 CCCCN=C(NCC(c1ccoc1)O)N(C)CC(c1c(F)cccc1F)NCC C1(C(N2CCCC(NC(C(CC)OC)=O)(CC)C2)=O)C2C3CC4C1C1C2CC3C41 c1(C(=O)NCC=C2CCN(C(CCC3CC(C)C3)=O)CC2)cc2cccnc2[nH]1 n1(CCC)cc(C(=O)N(C(CC)C(=O)NCCn2cncn2)C)nn1 N1(C(CC(COC)NC(c2cc[nH]n2)=O)=O)CC(C)(C)OCC1CO N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC(C)CC1CNC(=O)C(C)S(C)(=O)=O c1(SCC)ccc(CC(=O)NCC(CC)N(C(=O)CP(C)(C)=O)C)cc1 c1(C(=O)Nc2c(C)ccc(C(=O)OCC)c2)cc(Br)cc(OC)c1OC C1(C(=O)NCC2C(NC(=O)OC(C)(C)C)CC(F)(F)C2)CC2CCCCN2C1 C1(CN(C(=O)CSCCNC(=O)CCc2ccoc2)C)CCC(F)C1 CC(C)CC(CNC(=O)C(C)Cn1ccnc1)C(=O)N1CC(O)CC1C(C)C CC1C(=O)NCCCN1N(C)Cc1ccc(OC2CC2)cc1 C1(C(=O)NCCN(CCO)CC)CN(C(C2CCCC(O)C2)=O)CCC1(C)C C1(C(N2CCN(CC)C(=O)C2)=O)C2CCCC2CCN1Cc1ccccc1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCCC(CN(C(CSCCC)=O)C)C1 N1(C(c2cnc(S)nc2)=O)CCC2CN(C(c3scc4c3OCCO4)=O)CC2C1 c1(C(=O)NCCCC(C)(C)NC(C=C(CC)CC)=O)cc2c(C)cc(C)cc2[nH]1 c1(C(=O)NCC2(F)CC(NC(C(C)SC(C)C)=O)C2)cccc2oc(=N)[nH]c12 N1(C(CC(C)(C)C)=O)CCC(C2CC(NC(=O)CC3CC(n4cnnc4)C3)C2)C1 N12CCN(CC1)C(=O)NC(C)C2=O.C(=O)(CC(CC)SC)NC1C(C)(CC)C1 Cc1cc(C)c(C(=O)NC2CN(C(=O)Cc3cccs3)CCC2CO)c(=O)o1 c1(-c2onc(C(C)N(C)C)n2)nc(CC2CCC2)nn1-c1ccc(C(C)C)cc1 c1(C(N2CCC(C(N(CCC=C)CC)=O)CC2)=O)cccc(C#N)c1C C1(N(C)C(c2ccc(O)nc2)=O)CCCN(C(=O)C(C)(C)c2cccnc2)C1 C1(C(=O)NC2CCCC(NC(CC3C(C)OCC3)=O)C2)C2CC3CC(C2)CC1C3 N1(C(C2ON=C(CC)C2)=O)CCCC(C)(C(=O)N(C)CCc2cnc[nH]2)C1 C1(C(N2CC3C(NC(Cc4ccn(CC)n4)=O)(C3)C2)=O)CC2(CC(C)=NO2)C1 C(C(C(=O)NCCC1CCCN1C)C(C)(C)C)NC(c1c(F)ccc(C)n1)=O c1(NC(=O)NC2CC3CCC2(CNC(=O)C2CC2)C3)cccc(Cl)c1Cl C(=O)(CC(CSC)NC(C12CCN(CC1)C2)=O)NCCCN(CC)CC c1(C(=O)NCC2CCCN(C(C3(OC)CCCC3)=O)C2)ccc(=O)n2c1CCC2 N1(C(c2cccc(C)c2F)=O)CCN(C(=O)C(c2ccccc2)F)CC(O)C1 C1(NC(c2c(Cl)cc(C)nc2)=O)CC2CCC1C(NC(=O)CC(C)(C)C)C2 c1(NC(C(=O)NC(C)Cc2ccc(Br)s2)=O)cnn2c1CCCC2 c1(SCC#N)ccc(C(=O)NC2CCCC2C(=O)NOCC=CC(C)(C)C)cc1 C1(C(N(C)CCOCCO)=O)CC2CCC(C1)N2C(c1ccc(F)cc1O)=O C1(CC=C)(C(N2CCCC2C(C)NC(=O)C(CC)OCCOC)=O)CC=CC1 Cn1nnc2cc(C(N3CC4(C3)SCCC4NC(C3CC=CCC3)=O)=O)cnc12 c1(CC(=O)NCC2(NC(c3[nH]nnc3C3CC3)=O)CCC2)ccc2ccoc2c1 C1(C(=O)O)C[Si]2(CCCC2)CN1C(c1nc2n(c1Cl)CCCC2)=O c1(C(=O)NCC2CN(C(CC(C)OC)=O)C(C)(C)C2)nc2ncccn2n1 C1(C2CCN(C(C3(F)CC3)=O)CC2)(NC(c2ccc(NC)cc2Cl)=O)CC1 C1(C(N2CCC(C)(CNC(=O)CC(F)(F)F)C2)=O)(COC)CCCNS1(=O)=O c1(C(=O)NCC2C(NC(=O)CCc3csnn3)CC2)ccc(C(F)(F)F)o1 c1(NC(C(C)C2CCOC2)=O)cccc(NC(=O)C(=O)NCc2ccccc2)c1 C1(NC(c2c(Cl)cn(C)n2)=O)CC(O)CN(C(=O)CCSCC(N)=O)C1 N1(CC)CCN(CCCCNC2(C)CCCN2C(=O)OCC)CC1.C(C)(C)(C)O c1(SC)cc(N2CCOCC2)ncn1.C1(NC(=O)COC)CCN(C(=O)OC(C)(C)C)C1 N1(C(C2(OC)CCC2)=O)CCCC(C2CN(C(=O)CC3CCC=CCC3)C2)C1 c1(NC(c2c(-c3c(C)cncc3)ncs2)=O)ccc(C(F)(F)F)c(O)c1 c1(CNC(C2CCN(C(C3CC(=O)OC3)=O)C2)=O)ccccc1Br C(=O)(N=c1[nH]c(Cl)ncc1Br)C(=O)OC(C)(C)C.C1(CN)CC(CNC)CO1 c1(C(C(=O)NCC(CO)NC(C(C)(C)OCCC)=O)F)cccc(C)c1 CC(CS(C)(=O)=O)C(=O)N(C)CCOCCN(C)C(c1cnn(C)c1F)=O N1(C(CC2C(C)OCC2)=O)CC2CCC1CN2C(=O)C(C1CCOCC1)F CC1CCN(C(c2cnc3ccccn23)=O)CCN1c1nc(Cl)ncc1F C(CCC(=O)NCCCOCCNC(C1(Sc2nc[nH]n2)CC1)=O)N(C)C CC1CN(C(=O)C=CC2CCCC2)CC1(C)CNC(=O)C(O)CC1CC1 C1(CNC(C2CCC(C)(C)O2)=O)CN(C(=O)C#CC2CC2)CCCO1 C(=O)(C#CC(C)(C)C)N(C(C(C)C)C(=O)N(C)CC1CCCC2CC12)C CC1(C)CN(C(=O)CSc2n[nH]c(=N)s2)C1C1CCN(C(=O)C2=CCCO2)CC1 c1(NC(C(C=C)O)=O)cccc(CNC(=O)COCc2ncnn2C)c1 N1(CC)CCCC(C(=O)NCC(C2(O)CCN(C(C3(OC)CCC3)=O)C2)C)C1 CCC(CCC(=O)NC(c1cn(C)nn1)C(N1CCN(CCO)CC1)=O)OC C(=O)(C(CNC(=O)C(CCOC)NC(C)=O)C(C)C)N1CCN(CCC)CC1 C1(NC(CN(C(COC)=O)C)=O)CN(C(C2CNC(=O)CC2(C)C)=O)CC2(CC2)C1 CC1C(O)CC2CCC1N2C(=O)NC1(Cl)CC2CCC1O2 N1(C(CCCCC(C)(C)C)=O)CCC2CCCN(C(=O)CCSCC(N)=O)C2C1 N1(C(c2cc(C)c(O)nn2)=O)CCCC(C2CC2NC(=O)C#CC(C)(C)C)C1 n1(C(N(CCN(CC=C)C)C)=O)cc(C(=O)N(CC)Cc2ccco2)nn1 N1(C(C(C)=CC2CC2)=O)CCN(C(=O)C=CCOc2ccccc2)CC12CC2 c1(CC)nnc2n1CCCC2C(=O)NC1CCN(C(C2(C(=O)NC)CC2)=O)CC1 c1(NCC2(c3ccc(OC)nc3)CCCC2)nccc(=NCCC(C)c2cccs2)[nH]1 C=CCCCCC(=O)NCC(C1CC1)NC(C1(C(=O)N(C)C)CC1)=O C(=O)(CCS(=O)(=O)N(C)C)NCCC(C)NC(C1CCCCC1n1cccn1)=O N1(C(C=CC=CCC)=O)CC2CC(C)N(C(c3ccnc(F)c3OC)=O)C2C1 CCN=c1[nH]cc(C(=O)NCC2CCN(C(c3ncc(OC(C)C)cn3)=O)C2)s1 C(=O)(C1CCC(=O)c2cccn21)NCC(CNC(c1c(C)nc(C)c(C)n1)=O)C c1(CN2CCCC(c3nc(C(C)C)on3)C2)ccc(Br)c(Cl)c1F C=CC(C)N=c1[nH]c(N2CCC(C3CCS(=O)(=O)CC3)C2)nc2c1COC2 CCC1=NOC(CC(=O)NC(C)C=CC(=O)NCC(n2cccn2)C)C1 c1(COC)cn2cccc(C(=O)OCc3cccc(F)c3Cl)c2n1 C1(CC(=O)N(CC(C)C)CC(C)C)CCCN(C(C2CCC(=O)C2)=O)C1 C(c1cc(F)c(F)c(F)c1)=CC(N1C(C(=O)NCC(=C)C)C=CC1)=O C(CC(C(=O)N1CC(CNC(=O)Cc2nn(C)cc2Cl)C1)NC(C)=O)SC C(CS(=O)(=O)c1ccc(Br)cc1)NC1(CO)CCN(C)C1=O CCCC(C(=O)NCc1cccc(N2CCCC2)n1)OCC.N12CC(C1)C2=O C1(S(C)(=O)=O)(C(=O)NCC(CC)NC(C(C=CC)O)=O)CC1 c1(C(C)OC(c2cnc(C)s2)=O)ccc(F)cc1Cl N1(C(c2cc(OCC)n[nH]2)=O)CCCC2(CCN(C(C3CC(C)(F)C3)=O)C2)C1 C#CC1(NC(=O)COC2CN(C(c3cncc(C#N)c3)=O)C2)CCC(C)CC1 c1(C(=O)NC2CCCN(C(CCCC#C)=O)C2)ccc(CC)c(C#N)c1 N1(C(=O)C2=CCCO2)CC23CCCC2(C1)CN(C(c1ccc([N+](=O)[O-])cc1)=O)C3 N1(C(CN2CCC(OC)C2)=O)CCCC1(C)CNC(c1c[nH]c(=O)cn1)=O c1(C2(C(=O)OC(C(=C)Br)=O)COC2)cc(C)c(-c2ccccc2)o1 c1(N2CCC(NC(C3CCCO3)=O)C(F)C2)nc2ncc(Cl)cc2s1 C1(CC(=O)OC)C(N(C(C)C(=O)N(CCS(C)(=O)=O)C)C)CCCN1C(C)(C)C C(=O)(C(C)(C)C(=O)N1CCOCC1CCNC(c1cncc(Cl)c1Cl)=O)OCC c1(OC)c(O)cc(C(N2CC3(CC3)CC2C(N2CCC(C)(O)C2)=O)=O)cc1O C1(CSC)CN(C(c2sccc2Cl)C(=O)NCCC2(C)CC2)CCO1 N1(C(c2ccc(C(C)=O)o2)=O)CC2CCC1C1CN(C(=O)C(C)=CC3CC3)CC21 CC1(C)CCCCC(C(=O)NCC2COCCN2C(=O)C(Cl)=CCl)C1 n1(CC)cccc1C(=O)N(CC(=O)N(C1CN(C)C1)C)C Cc1cc(Cl)ccc1OC.C(C)(C)(CNC(=O)CC1CC=CC1)O.C1C(=O)NCC1 C1(CCC)CC(C(=O)NCC#CCNC(=O)CCC2SCCS2)C1 C1(C(N(CC(CC)NC(c2c(C(F)(F)F)cnn2C)=O)CC)=O)CN(C)C(=O)N1 C12(CC(=O)NC34CC(C3)N(C(C3(F)CC3)=O)C4)CCC(CC1)CC2 C(=O)(CC(C)(C)C(=O)NC1CN(C(c2ccn(C)n2)=O)CC1C(F)(F)F)OCC C(=O)(C(C)CCCCCC)N(C1CCN(C(C2(C=C)CCOCC2)=O)C1)CCO CC1CC(NC(c2cncn(C)c2=O)=O)CCN1C(c1ccc(CO)c(F)c1)=O c1(C(=O)NC2CCN(C(C3(C)CSC3)=O)CC2)cccc2[nH]ncc12 N1(C(C2(OC)CCC2)=O)CCC(C2CCN(C(C3CS(=O)(=O)C3)=O)CC2)C1 n1(CC(CC)O)cc(CC2CCCN2C(c2cnn(CCF)c2)=O)nn1 CC1CCN(C(c2cccc(CCN3CCCC3)c2)=O)CCC1(F)F C(CCCCCC(=O)NC1CC1c1cncs1)NC(CC1C(C)C(=O)CC1)=O N1(C(c2cnc(C)o2)=O)CCC(C2CCN(C(=O)C(F)(F)CO)C2)C1 S(=O)(=O)(c1ccc(CC#N)cc1)N(C1CCCCC1C)CC C=CCC(F)(F)C(=O)N1CC(CNC(=O)C(c2ccc(Cl)c(F)c2)O)C2(CC2)C1 C1(CCC(=O)N(CC(C)O)CC)CCN(C(c2csnn2)=O)C1 N1(C(C2(C)CCOCC2)=O)CC2(CCC(C(=O)NCC3(CO)CC4CC4C3)O2)C1 N1(C(C(C)(CO)NC(C2CC(CC)C2)=O)=O)CCC(C)OC(C)C1 c1(CNC(C2(CNC(C(c3ccn(C)c3)C)=O)CC2)=O)ccc(C#N)cn1 O=C1CN(S(=O)(=O)c2ccccc2[N+](=O)[O-])c2cc(Br)ccc2N1 C1(NC(CC(C)OC)=O)CCC12CCN(C(=O)C=Cc1ccc(=N)[nH]c1)CC2 Cc1cc(=NCCc2nnc(C)n2CCC)[nH]c(=NCc2ccc(N)cc2F)[nH]1 S(=O)(=O)(c1ccc(Cl)cn1)N(C(=O)C(F)(CN)CF)C c12ccc(nc1)oc2=O.c1(C(=O)NC2CC2CNCC(F)F)cn(C(F)F)cn1 CC(CCCNC(=O)C(C)(C1CC1)NC(=O)OC(C)(C)C)NCC(CC)C1CC1.C(Br)OC C(CC(O)C(=O)NCc1c[nH]nc1C(N1CC(CO)C1)=O)OC CC(C)CCC(O)C(=O)N1CCC(C(=O)NC(C)Cc2cccnc2)O1 N1(C(C(C)OCC(C)C)=O)CC2CC1CN2C(c1cc(N)cnc1Br)=O c1(SC)ccc(C=CC(N2CCCC2CNC(=O)Cc2cnccn2)=O)o1 c1(C(=O)NC2CCN(C(C3CC3CF)=O)C2)ccc(C(F)(F)CF)cc1 N1(C(Cc2nc(C)sc2)=O)CCC2C(NC(c3ccnc4c3CCC4)=O)C2CC1 CC1(C)CC1(O)C(N1CCC(CNC(=O)COC2(c3ccccc3)CCC2)C1)=O N1(C(CCC2CCC(=O)N2)=O)CC2CCC1CC2NC(c1cccc(O)n1)=O N1(C(CCC(C)NC(=O)CCc2nc(O)n[nH]2)=O)CC(F)(F)C(F)(F)C1 CN1CC(NC(c2ccc(CNC(C3(CO)CCCO3)=O)s2)=O)CC1=O c1(C(=O)NCC(C)NC(c2c[nH]nc2C2CCC2)=O)cc2c(F)cccc2s1 c1(NC(C2CN(C(=O)CCc3ccco3)CCC2(F)F)=O)ccc2c(c1)CCC2 CC(CCCCNC(C1CC1c1ccco1)=O)NC(c1cc(C2(O)COC2)on1)=O C1(C(N2CCC(CNC(C3(c4cccs4)CC3)=O)C2)=O)CCCC2(CC2)C1 c1(OC)cccc(C(N2CC3CC2C3CNc2csc(NC(=O)C(C)O)c2)=O)c1 N1(C(CC2ON=C(CC)C2)=O)CCCC(C(=O)NCC2(CCO)CC2)(CC)C1 N1(C(c2ccc(O)c(F)c2)=O)CCC2(CC1)CN(C(C13CCCCC1C3)=O)C2 C1(c2nn(C(C3CCC3)C)c(-c3cc(O)nn3C)n2)CCOC2(CCOCC2)C1 c1(CN(C(CC)(C)C)C(=O)C(C)N(c2ccccc2)C)ccc2c(c1)CC(=O)N2 CN1C(=O)c2ccccc2C1C(=O)N1CC(O)(CNC(c2ccnnc2O)=O)C1 N1(C(CCC(CC)OC)=O)CCC2CCN(C(c3n[nH]c4c3CCC4)=O)C2C1 Cc1cc(O)c(Cl)cc1C(=O)N(CCCCNC(=O)CN1CCCNS1(=O)=O)C Cc1cc(C(=O)NC2CC(NC(c3ccc(C(N)=O)o3)=O)C2)ccc1F N1(C(c2cc(F)c(Br)c(F)c2)C)CCC2(CC1)CC2N=c1[nH]cnc2cc(I)sc12 C=CC(C)(CC)C(=O)N1CC(O)(C(F)C(=O)NC(C2(O)CCC2)(C)C)C1 C1(CNC(C2(CC)CC2(F)F)=O)CCN(C(=O)CC2CCOC2(C)C)CC1 N1(C(C2(SCC)CC2)=O)CCC(NC(=O)CCc2ccc(Cl)cc2F)C(C)C1 Cc1cc(C(=O)NC2CCCC2CNC(=O)CSC2CC2)c(C)cn1 CC1CC(CO)CCN1C(=O)CC(C)(C)N(C)C(c1ccc(C2CC2)o1)=O CC1(C)CC(NC(c2ccnc(OC3CC3)c2)=O)CN1C(c1[nH]cnc1C#N)=O Cn1nnc2c(N3CCOC(CNC(C45CCCC4C5(F)F)=O)C3)ncnc12 N1(C(C2(CC#C)CCOC2)=O)CCC(C)(NC(=O)C(F)C2CCCC2)CC1 N1(C(C(=O)NCc2ccc(CC)o2)=O)CCCCC1c1ccccc1Br C1(C(F)(F)F)(C(=O)NCCOCCN(C(C2CC(SC)C2)=O)C)CC(C)(C)C1 c1(C(=O)NCC(=C2CN(C(=O)CNc3ccccn3)C2)F)ccnnc1Cl c1(C(c2nnnn2C2CC2)Nc2ccc(CC)cc2Br)cc(F)c(F)c(Cl)c1F C1(C(C)NC(C2(CO)CC(F)(F)C2)=O)CN(C(C2CC2(Cl)Cl)=O)CCO1 c1(C(=O)NC2CCC(C)(NC(C3CC4(C3)CC4F)=O)CC2)occ2c1CCCC2 N1(C(CC2CC(SCC)C2)=O)CCCC(C)(C)C1C(=O)NCCN1CCCOC1=O n1(CC)c(NC(C2CC(C)CN(C(=O)COCCF)C2)=O)nc2ccccc12 c1(-c2n(CC=C)nc(C3CCCO3)n2)cc2c(s1)CCSC2 N1(C(C(CCOC)OC)=O)CCCC(C(=O)Nc2cnsc2)CC1 C1(NC(c2c(C)coc2)=O)CN(C(=O)Cc2cn(C)cn2)CC1N=[N+]=[N-] c1(C(C)=O)ccc(C(=O)NCC(C)CNC(c2cc(C)oc2C(F)(F)F)=O)nn1 C#CC1CCCCN1C(c1ccnc(CNC(C2(SC)CC2)=O)c1)=O C1(C)(C(N(CCNC(C2N(CCC)CCCC2)=O)CC)=O)CCN(C(C)=O)CC1 C1(C(=O)NC2CCS(=O)(=O)C2)(NC(C2C(C)C2)=O)CCCCCC1 c1(C(=O)NCCC2CN(C(=O)CCC3CC3CC3CC3)C2)csc(=NC2CC2)[nH]1 O=C1CC2(C1)CC(C(=O)NCC1CC(C(=O)NCc3ncc(Cl)cn3)CCO1)C2 C(CC1=CCN(C(c2c[nH]nc2C)=O)CC1)NC(C1CCN(CC)C1)=O n1(CC(C)O)cc(C(N2CCC(NC(c3cc(N)cc(F)c3)=O)C2)=O)ccc1=O C12(NC(=O)CC3CC(=C4CC4)C3)CCCCCC1N(C(=O)CN1CC=CC1)CC2 C1(NC(c2cc(C)c(=O)[nH]c2)=O)CCN(C(c2cc3ccccc3[nH]2)=O)CC1C C1(F)(CNC(=O)CCC2CC2(Cl)Cl)CCN(C(C2(n3cnnn3)CC2)=O)C1 c1(C(N2CCC(N(C(c3nc(Cl)sc3C)=O)CC)C2)=O)ccc(C(C)=O)cc1F C(CCC(C)C(=O)NC1CC(C)CN(C(c2ccc(CC(N)=O)cc2)=O)C1)OC c1(OC)cccc(C(=O)N(CCCOCCNC(C2C3CCCOC23)=O)C)c1F N1(C(C2C(OC)(OC)CC2)=O)CCOCC1CC(N1CC=CCC1)=O C1(C(=O)N(C2CC2NC(C23CSCC2C3(F)F)=O)CCO)CCC(F)(F)CC1 C=CCC(C)(C)CC(=O)NCC(O)CCNC(=O)COc1cnn(C)c1 N1(C(CC(n2c(CC)ncc2)C)=O)CCC(CNC(c2cc(C)sn2)=O)CC1C CCS(=O)(=O)CC(=O)N1CC(NC(=O)CCc2ccccc2)CC(C)C1 N1(C(CC2CN(C(C)=O)C2)=O)CCN(C(=O)CS(N)(=O)=O)CC1CS(C)(=O)=O C1(NC(C23OC(C)C(C2)C3)=O)CN(C(=O)C=Cc2cnn(C)c2)CC2(CCC2)C1 Cc1cc(C(=O)N(C(C)CNC(=O)C(C)C2CCC2)C)ccc1OCC(F)(F)F N1(C(C(C)SC)=O)CCC2(COC(CNC(c3[nH]nc(C(F)(F)F)c3C)=O)C2)C1 c1(C(N2CCC(CCNC(c3nnn(C)c3N)=O)C2)=O)nn(C)c2c1CCCC2 c1(N2Cc3c(ccc(C)c3)C2)nc2cccc(F)c2c(=NCc2cc(C)[nH]n2)[nH]1 C(=O)(CC1OCc2ccccc21)NCCC(C)NC(C1=CCC(C)CC1)=O c1(C(=O)NCC(CCC)NC(=O)C(C)Cn2ccnc2)ccc(OCC)cc1 C1CCCC2(CC1)OCCC2N1Cc2ccccc2CC1 C1(CN(C(C(C)OCC(F)(F)F)=O)C)CN(C(=O)Cc2ccnn2C)CCO1 c1(C(N2CC(C)C(NC(=O)CCN3CCC3)CC2)=O)cc(Cl)cc(Cl)c1F C(CCCCC(=O)NC1CC(CCCNC(=O)C(C)CF)C1)NC(=O)OC(C)(C)C c1(C(N2CCN(C3CCN(C(CCC)=O)CC3)CC2)=O)cc2sc(C)cc2s1 c1(C(N2CC(OCCNC(=O)CC3CC=CC3)C2)=O)ccc(C2CC2)nc1O c1(C(=O)NCCC2(O)CCCN(C(C(C)S(C)(=O)=O)=O)C2)ccc2c(c1)OCO2 C(=O)(CC(C)C(C)(C)NC(=O)C=C(C)COC)N1CCC(CC=C)C1 c1(C(=O)NC2(C)CCCN(C(c3nccc(N)c3Cl)=O)C2)nccc2[nH]ccc12 C1(C(=O)NC2CN(C(C)(C)C)C2)CCC(=O)N1.C12(OC)CC1C(=O)NC2 C1(CCC#N)(C(=O)NCCCN(C(c2cc(OCC)no2)=O)CC)CCCC1 N1(C(CC2(OC)CCC2)=O)CCC(C(C)NC(C2CC2C(F)(F)F)=O)CC1 C(=O)(C(C)CC(N)=O)NCC(C)=CC(=O)NC1C(=O)OCC1CO C(C)(C)(CC(=O)NCC1(C)CCN(C(=O)CC2CC(F)(F)C2)C1)OC C12C3CC4C(C3)C14C(=O)N2.O=C(CC(=O)NCC1CC1c1ccco1)N.C(O)=C C=CC1(C(N2CCSCC2)=O)CCN(C(c2csnn2)=O)CC1 C(CC(=O)N(CCN(C(c1csc(C)c1)=O)CC)CC)(C(C)C)OCC c1(C(=O)NCC(CO)NC(C(c2cn(C)nc2)(F)F)=O)cccc(C2CC2)c1 N1(C(c2ccc(SC)s2)=O)CCC2CN(C(=O)C(c3cccnc3)C)CC2CC1 c1(C(=O)NCC2(C(N)=O)CN(C(C3CCC(C)O3)=O)C2)coc2ccc(O)cc12 N1(C(C2(C)C(CC)CCC2)=O)CC(NC(c2cnn(C)c2)=O)C(C)(C)C1 N1(C(C2(C=C)CCC2)=O)CCCCC(CNC(C2CCCC(O)C2)=O)C1 n1(CC(=O)N(C(C)CNC(C2CC2(F)F)=O)C)cnc2c1CCCC2 c1(OC)nc(C(N2CCN(C(c3cc(OC)ccc3F)=O)C3CC23)=O)cc(O)n1 c1(CC(N2C(C(N3CCC(C)(N(C)C)C3)=O)C(O)CC2)=O)cccc(Br)c1F C(CCC(C)(C)C(=O)N(C)CC1CC1C)NC(C=CCCC)=O C(=O)(C(C)(C)C(=O)N(C)C)NCC(C)(C1CC1)NC(C(CC)CC1CCCC1)=O c1(NC(C(CCOCC)NC(=O)CC2(C(F)F)CC2)=O)ccc(CC)c(C)c1 N#Cc1cc(C(N2CC(NC(c3cncs3)=O)C3(CC3)C2)=O)ccc1O C(CCCCCN(C)C(C1CC1CCC)=O)NC(C1(CC#C)CCCO1)=O N1(C(C(=O)N(C2(C)CC2)C)C2CC2C2OCCO2)CCC(F)(F)C(CO)C1 c1(CC)cc(C(=O)NCCCCCNC(=O)CCc2nc[nH]n2)nn1CCO c1(CNC(C2(C3N(C(CCC=C)=O)CC3)CC2)=O)ccc(Cl)c(OC)c1 N1(C(CN(C(=O)C(c2cccnc2)C)CC#C)=O)CCC(C2CC2)CC1 C1(NCC2(CC(=O)OCC)CC2)CCCN(C(C2CN(C)CC2C(F)(F)F)=O)C1 N1(C(C=CCC)=O)CCN(C(=O)CCC(C)(C)C)CC1C(C)C C1(N2CCOCC2)(C(N2CC(CN(C(C(C)OC(C)(C)C)=O)C)C2)=O)CCCC1 N1(C(CCC)=O)CC(NC(=O)CCCCNC(c2ccccc2Cl)=O)C(F)C1 C1(C(N2CC(NC(C=CCOC)=O)C3(C2)CC3)=O)OC(C)(C)OC1(C)C C1(CNC(c2cnc3[nH]ccnc2-3)=O)CCC2(CN(C(c3cccnc3)=O)C2)O1 C(=O)(CCCCCF)N1CCC(OCC(N(OCCCC)C)=O)C1 n1(CC(N2CC(NC(C(C)SC)=O)C(C3CC3)C2)=O)c(=O)cnc2ccccc12 C(=O)(C(C)(C)C(C)(F)F)N(CC(C)C(=O)NC(C)C(=O)NO)C N1(C(c2ncn(C(C)C)n2)=O)CCN(C(C2CC(CC(F)F)C2)=O)CC1C(C)C C1(F)(NC(C(C=C)c2ccccc2)=O)CCS(=O)(=O)C1.C12CCC(C1)CNC2=O c1(C(=O)NCCN(C(=O)COCC(F)(F)F)CCC)c(C)ccc(Br)c1C C1(C(N2CCCC(C)C2)=O)N(C(=O)CN2CCCC2=O)CC12CCCC2 C12(C(N(CC=C)CCOC)=O)CCC(CN(C(=O)CC3CC(C)C3)C1)C2 N1(C(c2cc(-c3nc(C)sc3)sc2)=O)CCC(O)(C(C)CNC(=O)OC(C)(C)C)C1 Cc1cnc(N)c(C(=O)NC2CCOCC2NC(=O)Cc2coc(C)n2)c1 C1(O)(C(N2CCC(CCN(C(=O)C(F)C3CCC3)C)CC2)=O)CCC(C)(C)CC1 C12(NC(C(F)=CCC)=O)CC(CNC(=O)CC(O)C3CCCC3)(C1)OC2(C)C C12CCC(CC1)NC(=O)C1OCC(C1)C(=O)OCC1CCC(C1)C(=O)N2.CC.SC C1(CNC(CN2CC(C)C2)=O)C(NC(=O)C(c2ccccc2)N(C)C)CC1O c1(CCCN(c2ccccn2)C(=O)NCc2c(C)scn2)cccc(F)c1 C1(SCC)CCC(N(C(=O)CCCc2cnn[nH]2)C(C)=O)C1 c1(C(N2C(CCNC(=O)C(c3ccccc3Cl)CO)CCC2)=O)ncncc1F c1(OCC)nc(N(CC(C)NC(c2ccc(C(C)(C)C)cc2)=O)C)ncc1C N1(C(c2cc(C(C)C)on2)=O)CC(CCNC(=O)C(C)=C2CC2)OC(C)C1 c1(OCC)cc(N2CCC(C)(CNC(C3(C)CS(=O)(=O)C3)=O)C2)nc(C)n1 CN1CC(C(N2CCC2(C)CC(=O)NCc2ccc(CO)o2)=O)CCC1=O C1(NS(CC)(=O)=O)CN(C(=O)C(C)(C)CC#N)CC1(F)F Cc1ccc(C(=O)NCCc2n[nH]cc2C(=O)NC2CC2(C)C(F)F)nc1O N1(C(C(C)(CO)NC(C2CCC3(CC3)C2)=O)=O)CCn2ccnc2C1 C1(CC(=O)NC(CC=C)CNC(c2ccnc(Cl)c2O)=O)CC2(CCCC2)CO1 N1(CC2CN(C(CCC)=O)C2)CCN(C(C2(COC)CCCCO2)=O)CC1 C1(CCCCC)CCCN(C(c2ccc(OC(C)C(=O)O)cc2)=O)C1 c1(C(=O)NC2C(C)N(C(=O)C(CCO)N(C)C)CC2)[nH]nc2ncccc12 C(CC(=O)NC1C(NC(=O)CN(C(=O)COC)C)OCC1)(OCC)OC.C1(OC)CC1 c1(NCC)cncc(C(=O)NC23CC2CN(C(c2ccncc2Cl)=O)C3)c1 c1(C(=O)NC2CCCN(Cc3cccc(C(F)(F)F)c3)C2)cc(Br)c(F)cc1F N=c1[nH]c(=NCCn2cccn2)[nH]c(=NC2CCN(C(=O)N(C)C)C2)[nH]1 c1(C(=O)NCC(C)(CO)NC(c2c(CC)nc(C)[nH]2)=O)cccc2c1ncn2C Cc1cnc(C(N2CCC(CCN(C(=O)Cc3cnccn3)C)CC2)=O)cc1C c1(NC(c2cncnc2)=O)cnc(Cl)cc1C(N1CCSCC1)=O c1(C(N2CC3CN(c4ncc(OC)cn4)CC32)=O)ccc(C#N)c(F)c1 c1(NC(c2c(F)ccc(Cl)c2Cl)=O)cc2c(cc1Br)OCCO2 C(CC(C(C)(C)C)NC(=O)CCc1c(Cl)cccc1Cl)N(C)C N1(C(C(CC(C)(C)NC(=O)CCc2cn[nH]c2)F)=O)CCC2CCCC2CC1 C(C(C(=O)N1CC(C)(C)CC1CNC(=O)C(O)C1CCCC1)C(F)(F)F)OC c1(CCNC(CC(C)N(C(C(C=C)O)=O)C)=O)ccc(C)nc1 C=CCCCCCC(=O)N1CCN(C(c2coc(Cl)n2)=O)C(c2ccncc2)C1 Cc1cnncc1C(N1CC(N(C(=O)CN2CC(F)(F)C2)CCO)C1)=O C1(CC(=O)NCCCCNC(c2cnsc2)=O)CCCC(O)C1 C(=O)(CCCCC(N)=O)NCCC1CC(OC)CN1C(c1cn2c(n1)CCC2)=O N1(C(c2c(CCC)nns2)=O)CCCC(NC(C23CC(CO2)C3)=O)C1C C1(C(C)C)CN(C(=O)CN(C)C)CCCN1C(=O)C(CO)N(C)Cc1nncn1C c1(C(=O)NC2C(NC(c3cc(CC)on3)=O)CCC2)noc(C)c1Br C1(NC(CCc2ccn(C)n2)=O)CC2CN(C(C3CC(O)C3(C)C)=O)CC12 C(=O)(C(C)C(C)NC(C1(C)CCC(=O)N1)=O)NCC1CCN(C(C)=O)C1 c1(C(=O)NCCN(C(C(CC(C)C)(F)F)=O)C2CCCC2)nccc(Cl)c1Cl Cc1cnc(CN2CCCC(O)(CNC(C3C4CCC(C4)C3C)=O)C2)cc1Br C(=O)(C(C(=O)N(C(C)C(=O)N(C1CCCC1(C)O)C)C1CC1)OC)OCC C1(NC(=O)C2=CCOC2)CCSC12CN(C(c1ccc(O)cc1C(F)(F)F)=O)C2 c1(C(N2CCC(CNC(C(CC=C)N(C)C)=O)C2)=O)ccnc(F)c1OC Cc1csc(CC(N2CCCC2CN(C)C(c2cnn(CCO)c2)=O)=O)n1 C#CCCCCC(c1nnnn1C1CCC1)NC1CCC(CNS(C)(=O)=O)CC1 c1(C(=O)NC2C=CCC(C(=O)NC3(CC=C)CC3)C2)cnc2ccccn12 c1(NC)cnncc1C(=O)NCC1(NC(=O)C(=CC2CCCCC2)F)CC1 S(=O)(=O)(c1c[nH]c2ncc(Br)cc12)N1CCC(OC)CC1 Cc1ncc(C(=O)NCC23CC(CN2C(C2CC(N(C)C)C2)=O)C3)c(C2CC2)n1 C1(NC(c2c(COC)scc2)=O)CC(C)N(C(=O)C=C(C)c2cccs2)C1 Cc1cc(C(N2CC(C(=O)N(C3CC=CC3)C)OC(C)C2)=O)c(O)nn1 C(CCCC(=O)N1CCC(C(F)C(=O)NOCC(C)(C)C)C1)(OC)OC.C=O c1(C(=O)NC(CC(C)NC(c2cc(C)c(C)o2)=O)C)ncc(C(N)=O)cc1Cl C1(C(=O)NCC=CCCC)CCCCC1CNC(C1CN(C)C1)=O c1(CC(=O)NCCOC2CCN(C(CNC(CC)=O)=O)C2)ccc(Cl)c(C)c1 C#CCC(C)(C(=O)NCC1CC1(F)F)NC(=O)CCOC1COC1 C1(C(=O)NCC(C(C)C)NC(CC2(C(=O)OC)CCC2)=O)CC2C(C1)C2(C)C C(C)(N=c1cccn[nH]1)C1(S(CC)(=O)=O)CC1 Cc1cc(C)c(C(=O)NC(C)(C)C(C)NC(C23CC4CC2C3C4)=O)o1 CN1CCC(C(=O)NCC(C2CCN(C(=O)Cc3cc(Cl)cs3)CC2)(C)O)C1=O N(C(=NCCCF)NC(C(C)C)c1cccs1)C(C1CCCCC1)C C12(CNC(=O)C=C3CN4CCC3CC4)CC(CO1)N(C(C13CC4CC1C3C4)=O)C2 C1(CC(N2CC(c3cn(CCOC)nn3)C(O)C2)=O)COc2ccccc2O1 C1(NC(c2cnc(-c3cccs3)s2)=O)CCN(C(=O)C2CC2)CC12CCC2 c1(NC(=O)CN(C(C2N(S(CC)(=O)=O)CC(F)C2)=O)C2CC2)cc(Cl)ccc1Cl c1(OC)ccc(C(=O)NCC(C2CC2)NC(=O)CC2CC3(CC3)CO2)c(C)n1 CCCCC(=O)C(=O)NC1(C)CC(NC(=O)CCc2ccccc2C(=O)NC)C1 Cn1ncc2c1CC(C(N1CCCC(CCNC(=O)C#CC(C)(C)C)C1)=O)CC2 Cc1nc(N2CCC(C)C(NC(=O)C(=O)NCC3CC3)C2C)c(F)c(C)n1 c1(NC(C2(C)CCN(Cc3c(Cl)cc(Cl)cc3Cl)C2)=O)nccn2c(Br)cnc12 C1(CNC(C2CN(C(C)=O)C2)=O)CN(C(C23CCOC(C)(C2)C3)=O)CCN1C C1(NC(c2cn(CC(CC)O)nn2)=O)CCN(c2cc(Cl)nc(C)n2)CC1F C1(C#N)(C(=O)N(CC(C)(C2CC2)NC(=O)CCCS(N)(=O)=O)C2CC2)CC2C=CC1C2.C N1(C(=O)NC(c2cccc(C)n2)C2CC2)CCN(S(=O)(=O)N(C)C)CC1 C1(CNC(C(C)N(C)C)=O)(NC(c2ccc3oncc3c2)=O)CC2CCC1CC2 C#CCC(C(=O)N(CC(C)O)CCNC(=O)Cn1ncc(Cl)c1C)C1CC1 C=CCCCC(C(=O)NCCCCCCO)NC(=O)COC1CCCCC1 CCC(CC(F)F)C(=O)N(CC(C)(C)CNC(c1ccc(Br)c(C)c1)=O)C c1(C(=O)NC2CCN(C(C(c3cccnc3)OC)=O)C2)coc2c1C(=O)CCC2 C1(C#CC(=O)N2CCCC(Nc3cc(O)nc(O)n3)C2)(CC)COC1 C1(C(N2CCC(CCF)C2)=O)CCN(CC(O)CO)CC1.c1cccc(Cl)c1 CN1CCC(C(=O)NCC2CCC(C(=O)Nc3csc(Br)c3)CC2)CC1 c1(C(N2CCCC(N(C(=O)CC3C=CCC3)CC)C2)=O)cc(C)c(=O)n(C)c1 C(C)(C(=O)NC1CC(C(C)C)C1)NC(CN(C(COC)=O)C)=O Cc1nccc(CCC(=O)NC2CCN(C(c3ccc[nH]3)=O)C2C(C)(C)C)n1 C(=O)(CS(=O)(=O)C1CC1)NCC(n1cc(CN2CCN(C)CC2)nn1)(C)C n1(CCCC)ccc(=NC(C)(CC(OC)OC)c2nnnn2C)[nH]1 c1(OC)cccc(CNC2(CCC(=O)NCCC3CCCC(C)C3)CCC2)n1 N1(C(CC(=C)C)=O)CCC2(CCOC2)C(CNC(C2CCSC2)=O)C1 C1(CNC(=O)Nc2sc(Cl)cc2Br)CCCC(C(F)(F)F)C1 C1(COC)(NC(=O)CN(CC(C)C)C(C2SCC=C2C)=O)CCSC1 C1(NC(CCc2ccn(C)c2)=O)CC2CC1N(C(=O)CN1CCC(F)(F)C1)C2 CCC(CC)C(=O)N1CCCC(CC(=O)N(C)OCc2ccccc2)C1 C1(NC(c2cnc(CC)s2)=O)CC2CN(C(C3CN(C4CCOC4)C3)=O)CC2C1 C1(C(=O)NCc2nc(CO)n[nH]2)CN(C(c2c[nH]c(=S)cn2)=O)CCO1 c1(C(=O)NCC2CCN(C(C3COC(=O)O3)=O)C2)cnc2ccoc2c1 c1(N2CCC(C)C(C)(C)C2)nc(N(C)CCC2CCCO2)nc2c1CC(C)CC2 c1(C(=O)NCCC2CCN(C(Cc3ncn(C)c3)=O)CC2)cnc2ccccn12 C(=O)(C(O)C(C)(C)C)N1CCC(N(C(CC(C)O)=O)CCO)C1 N1(C(C(CCC)F)=O)CC(CNC(c2ccc(NC(C)=O)cc2Cl)=O)C(C)(C)C1 c1(C(=O)NCC(CN(C(C(C2CCCO2)OC)=O)C)C)cc2c(F)cccc2s1 C1(C(N(C2CC(NC(c3[nH]cc(C(C)=O)c3)=O)C2)C)=O)CC(=O)NC(C)C1 N1(CC#C)CCC(C(=O)OC(C(F)(F)F)C2CC2(C)C)CC1 C(=O)(C(C)CC(C)(C)C)NC1CC2CN(C(c3c(CCC)[nH]cc3)=O)C1C2 C1(C(=O)NC2CCN(C(C34CCCC3OCC4)=O)CC2)CC2(CCC2)CO1 C1(C(NOC)=O)CC(NC(c2ccsc2C)=O)CO1 N1(C(C(C)N(CC)CC)=O)CCCC(NC(=O)CCNC(=O)C=CCl)C1 C(=O)(CCC1=CCCCC1)NCCC(C)NC(c1cc(F)c(C(F)F)cc1F)=O N1(C(C#CCNC(c2cccc(O)n2)=O)=O)CCC2(CCCCC2)C1 c1(C(=O)NC2C(CNC(CC(=O)OC)=O)CC2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 C1(C)(c2cn(CC)nn2)CCN(c2ccc(CC(=O)NC(CC)C)cc2F)CC1 CCC(C(=O)NCCOCC(=O)NC1CCn2cncc2C1)C(F)(F)F N1(C(C2CCN(C)C2)=O)C2CC1CN(C(c1cncc(-n3ccnc3)c1)=O)C2 C(CCC)(C(=O)N1CCC(C2CCCN2C(C2(COC)CC2)=O)C1)=CCC c1(C(=O)NCC(C2CCC2)NC(C2C(C=C)CC2)=O)ccnc(C2CCC2)c1 C#Cc1cccc(CC(=O)NCCN(C(=O)C(C)(C)N(C)CCC)C)c1 c1(C(N(CCNC(=O)CCc2conc2C)CC)=O)ccc(N)c(Cl)n1 N1(C(C(C)=CC)=O)CC2CN(C(c3ccc(-c4ccc(Cl)cc4)s3)=O)CC2C1 c1(N2CCC(CC=C)(N(C(=O)C(O)C(C)CC)CC)C2)nn2cc(C)nc2s1 Cc1nnc(NCC2CCCC(NC(c3nn(C)cc3Cl)=O)C2)c(C#N)c1C N1(C(C(CC)C#N)=O)CCC2(CC1)CN(C(=O)CCc1cc(C)on1)C2 N1(C(C(OCC)OCC)=O)CCCC(n2cc(CC(O)C3CC3)nn2)CC1 C1(N(C(=O)Cc2nc(Cl)cs2)CC2CC2)CCCN(C(=O)COCC(F)(F)F)C1 CCCCC(O)C(=O)NCC1C=CCN1C(=O)CSc1ccnc(C(F)(F)F)c1 C#CCC(CC#C)NC(=O)CC1CCN(C(=O)CC(C)n2ccnc2)CC1 CN1C(=O)COC(CNC(=O)C(C2CCC(F)(F)CC2)F)C1c1cnn(C)c1 CC(C(=O)NCCC1CN(C(C2(CCS(N)(=O)=O)CCC2)=O)CCO1)C(F)F C1(C(=O)NC2CCN(C(CCc3ccn(C)n3)=O)C2)CC(C)(C)OC1(C)C c1(NCCC2CCCN(C(c3cc4n(n3)CCO4)=O)C2)ccc(Br)cc1[N+](=O)[O-] c1(C(=O)NC2CC3CC(NC(C4C(C#N)C4)=O)C2C3)ccc2[nH]ccc2n1 C(=O)(C(CCCOC)NC(=O)CCN(C)CCO)NC(CCC=CC)C N1(CC(=O)NCC2C(NC(C34CC(C)C3C4)=O)CC2)CCCCCC1 C1(C(=O)NCC2CCCN2C(=O)C(F)n2cccn2)CC12CCCC2 C1(CC(=O)NC(C=C)CO)CN(C(=O)CC2CC3C=CC2C3)CC12CC2 C1(CN(C(=O)CCC2CC2)C)CN(C(=O)C(C)(C)CN2CCN(C)CC2)CCO1 CCCC(C(O)C(=O)NCc1cnc(C)o1)NC(=O)C(CC(C)C)OC C1(CCC(=O)NCC#CC(=O)OC)CCCN(C(=O)CCC2CCCC2)C1 N1(C(=O)CSc2ccncc2)CC(C2CN(C(C3CC4(CCC4)C3)=O)C2)C1 O=C1CCC(N2CCC(N3CCC(C(O)C(F)(F)F)CC3)C2=O)CN1 CC1C2CCCCC2CN1C(=O)CC(CC1CC1)NC(=O)Cc1cc[nH]c1 C1(C(=O)NCC(C)CNC(c2cc(F)cc(Cl)c2O)=O)CCC2(CCC2)CC1 C1(C(N(C)Cc2cc(C(C)(C)C)no2)=O)CC2(CCC(=O)CC2)C1 CC1CN(C(C2CCC(=O)N(C3CC3)C2)=O)CCC1NC(C1CCS(=O)(=O)C1)=O C1(=O)C(C(C)C)N1.c1(CC(=O)NCCN(C(=O)C(F)(F)F)CC)ncc(C)s1 CC1CN(C(c2cc3[nH]ccc3s2)=O)CCN1C(c1csc(C2CC2)n1)=O C1(C(N(CCC#C)CC)=O)CC(F)CCN1C(C1CCC(C)(C)C1)=O C(=O)(C1=C2CCN=C2NC=C1)N1C2C(CNC(c3c(C)c(Cl)ccc3)=O)C(C2)C1 CCCCCC(O)C(=O)NCCCCCC1CCN(C(=O)C=C(C)Cl)CC1 c1(C(N2CCC(CNC(c3ccc(CC)s3)=O)C2)=O)cc(Cl)n(C)n1 C12=NC(=NC34CCCC3CN(C4)C1=O)SN2.c1(COC)cn2c(n1)CC(C)CC2 c1(C(=O)NC2C(CC(C)C)CNCC2)sc2c(c1I)CNC2 C#CCCCCCC(=O)N(CC(C)(C)CNC(=O)CC1CCCNC1=O)CC c1(OC)cccc(C2N3CCC(C3)CNC2=O)c1F.C(CC#N)OCC C1(CCNC(CCOCCCOC)=O)CCCCN1C(=O)CC1CCC1(C)C N1(C(=O)NCCCN(C(C)C)C)CCC(c2nc(C(F)(F)F)cs2)CC1 C1(NC(c2c(C(C)C)onc2)=O)CCCC(NC(c2occc2F)=O)C1 c1(OCC)cc2c(cc1F)N(C(=O)C(=O)N(CCC1=CCCCC1)C)CCC2 CCC(CC)CC(=O)N(C1CCN(C(c2ccc(C(F)F)nc2)=O)CC1)CC C(C(C)C(=O)NCC(C)CNC(=O)CNC(C1CCCC1)=O)SC C(=O)(CCC(CC)NC(=O)CCc1cncs1)N(CC(=O)N(CC)CC)C C1(NC(C(C2=NOC3CC23)NCC2C(C)(C)C2(C)C)=O)Cc2ccc(Br)cc2C1 c1(C(=O)NCC2N(C(C(C3CC3)SC)=O)CCC2)n[nH]c(C)c1O c1(C(N2CC(OCC(=O)NCC(C#C)C)C2)=O)nonc1C C#CC1(C(=O)NC2C3CCCOC23)CN(C(=O)CC2CCCSC2)C1 Cc1nn(C)c(CNc2cc(OC(C)C(=O)O)cc(F)c2)c1I CN1CC(O)CC1(C)C(N1CCC(Cn2cc(C3CCC=CO3)nn2)CC1)=O N1(C(c2cc[nH]c2C2CC2)=O)CC2CCN(C(c3n[nH]c4c3COCC4)=O)C2C1 N1(C(c2c(C)cc[nH]2)=O)CCC(CN(C(C2CC2CC(C)C)=O)C2CC2)CC1 c12conc1C(C)N(C)C(=O)N1CC2C1.C(=O)(C1CC1)OC c1(C(N2CC(NC(CCCCC#C)=O)C(O)C2)=O)cc2sc(Cl)cc2[nH]1 C(=O)(CC(O)CC(C)(C)C)NCC(CN(C(=O)COC1CC1)C)(C)C C12CSCCN1C(=O)CN(C)C(=O)CC(=O)NCC2.Cc1nc(SC(C)C)n[nH]1 C(=O)(CCC(C(C)C)NC(=O)C=CC(C)C)NCc1cccc(C)c1F c1(C(=O)NCCCCCN(C(=O)CC2C=CCCC2)C)cc2c(s1)CCC2 N1(C(C2CCN(C)C2)=O)CC2CC1CCC2NC(c1nn(C)c2c1CCC2)=O C(CN=c1[nH]c(N2CCC(N=[N+]=[N-])C2)nc2c1CSC2)N(C(C)(C)C)C C1(NC(Cc2n(C)ncc2)=O)CCOC(C(=O)NCC2CCCCC2O)C1 Cc1nc(Cl)c(NC(=O)C(C)NC(=O)CN2CC3CCC(C2)C3N)c(C)c1C C1(NC(c2ccc(OC)nc2Cl)=O)COC2(C1)CN(C(=O)Cn1ccc(C)n1)C2 Cn1c(O)nc2ccc(NC(N3CC(F)(F)C4(CC(O)C4)C3)=O)cc12 C1(NC(=O)COc2cn[nH]c2)CCCN(C(c2cccc(C(F)(F)F)c2)=O)C1 c1(C(C(=O)NCCCCCC)N(CC(C2CCC2)OC)C)cnc(C)cn1 C1(NC(C2(C)CCC(=O)N2)=O)CCN(C(=O)C(F)(F)C(O)C2CC2)CC1O C(=O)(C(CN=c1ccc(S(C)(=O)=O)c[nH]1)c1cccc(Cl)c1)NC N1(C(C(C(C)C)O)=O)CCN(C(c2ccccn2)=O)C(C#N)C1 C(=O)(C(CC(C)C)NCC(C)C(=O)OCC)OC(C)(C)C CC(F)(F)CC(=O)NCC1CC(NC(=O)CN2CCNC(=O)C2)C1(C)C C1(C(=O)NCCCSCC)CN(C(c2ccnc(CC)c2)=O)CC1F CC(C(F)(F)C(F)(F)F)=CC(=O)NC(C)(C)C(C)NC(=O)C(=CC1CCCC1)C c1(C(=O)NC2CC3CC2N(C(C2CCCC2)=O)C3)cnc2c(F)cccc2c1 N1(C(C2CCCS2)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)C(c2ccncc2)C1 CC1CC(=O)NCC1C(=O)N(CC(C)(C)C(=O)NCC1C2CCCC12)C c1(C(N2C3CC(NC(CC(C)(C)O)=O)C(C3)C2)=O)cc2ccccc2o1 C#Cc1ncc(F)cc1NC(N1CCC(O)C1c1ccccc1C)=O CC1CC(CC(N2CC(F)(CNC(=O)Cc3ccccc3F)C2)=O)CC(C)(C)C1 C=CC(C)(CC)C(=O)N(CCCCN(C)C(c1c(OC)cccc1F)=O)C Cc1ccc(C=CC(=O)NCC2CCCCN2C(C2(CO)CC2(F)F)=O)o1 c1(C(N2CC(OCCNC(=O)CC3CCCOCC3)C2)=O)cccc2occc12 c1(OC)ccnc(C(=O)NCC(C)(C)NC(c2n[nH]c(C)c2O)=O)c1F C1(NC(C2(OCC)CC2)=O)CC2CC(NC(C3CN(C)C3)=O)CC12 c1(CCC(=O)NCC2N(C(C3CCC(C)O3)=O)C3C(C2)C3)ccc(Cl)cc1F N1(C(C2CCOC2)=O)CCCC2CN(C(C3(C4CCCO4)CCC3)=O)CCC12 C1(C(N(CCOCCOC)C)=O)CC12CCN(C(=O)C(C)CC(F)F)CC2 CC1(C)CCOC1CC(=O)NCc1cccc(C(=O)NC2CC(C)(O)C2)n1 c1(C(N2C(C(N3CC(C)(CC)C3)=O)CSC2)=O)cccc(F)c1 N1(C(C2N(C(CSC(=N)N)=O)CCC=C2)=O)CC(O)C(O)C1CO C1(C(=O)NCC(=O)NCc2cn(CC(=O)NC)nn2)CCC(CO)CC1 C1(C(=O)NCC(C)(C)OCCNC(c2[nH]ccc2C2CC2)=O)CC2CCC2C1 C12(C(=O)NC(c3nnc(O)o3)C)CCCC1N(C(=O)CCCC1CCCO1)CC2 CCCCC(CNC(c1ccnc(C)c1)=O)NC(c1cc(Br)sc1C)=O N1(C(C(=O)NC(CCC=C)C(=O)OC)=O)CCCC2CN(C)CCC12 c1(NC(CN2CCCC(OCCC)CC2)=O)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NCC2C(NC(C3C(C=C)OCCC3)=O)C2)[nH]c2ccccc2c1C C1(NC(=O)CC=CCNC(=O)CC2CCC(=O)N2)CCc2nncn2C1 N1(C(C(=O)NCCOCC)C2CC2Cl)CCCC1C1(C)CC1 C1(NC(c2n(CC#C)ccc2)=O)CCN(C(c2cc(C(C)C)nn2C)=O)C(C)C1 C1(C(=O)NC2(CC=C)CCC2)(NC(=O)COc2cc(C)on2)CCSC1 c1(C(=O)NCC23N(C(c4ccc(C)c(C)n4)=O)CC(C2)C3)c(C)nc2sccn12 N1(C(c2c(OC)cc3c(c2)CCC3)=O)C2CCC1CC1(C2)CC1(F)F c1(OC)cccc(C)c1C(N1CC2CC1CC2NC(c1ccn(C)n1)=O)=O C1(N(C(=O)CCN(C(=O)CC2(N(C)C)CC2)C2CC2)C)CCCC1(C)O c1(C(=O)NC(c2cn(Cc3nc(C(N)=O)cs3)nn2)C)cc2cnn(C)c2s1 c1(C(=O)NCC(CN(C(C2NC(=O)CC(C)C2)=O)C)O)cnn2c1N(C)CC2 CCCS(=O)(=O)CC(=O)N(CCCNC(c1cccc2cncn12)=O)CCO CC(C)CC(C(=O)N1CC2CCN(C(c3coc(CO)c3)=O)C2C1)C(C)C N1(C(C(=O)NC(C)C)=O)CC2(CCC(NC(c3nn(C)c4c3CCC4)=O)C2)C1 N1(C(Cc2c(C)n[nH]c2)=O)CC(F)CC1C(=O)NCC1CCOC1C N1(C(C(COC)N(C)C)=O)C(CC(N2CC(F)(C3CC3)C2)=O)C2CCCC12 C1(c2[nH]cc(C(=O)OC(C)(C)C)n2)CCN(C(=O)COC2CCCC2O)CC1 C1(C(=O)NC2(CCCNC(c3cn(C(C)C)nn3)=O)CC2)CC(C)CC(=O)N1 N1(C(c2cc(C)no2)=O)CC2(CC(NC(=O)C=C3CCCC3)CO2)C1 CCC(C)CCCC(=O)NCC(O)CCNC(c1cscc1C#N)=O c1(C(N2C(CNC(C(CC=CCC)C)=O)CCC2)=O)cnc(C)[nH]c1=N N1(CCC(N2CCCC(c3ncc(N(C)CC)s3)C2)=O)CCCC2(CC2)C1 CCCC(CC(C)C)C(=O)NC1CCN(C(=O)Cc2ccc(OC(C)=O)cc2)C1 N1(C(C(C(C)(C)C)N(C)C)=O)CC2C(C1)CS(=O)(=O)C2.c12cn(nn1)CC2 C1(C(N(CC(C)N(C)C(c2cc(C3CCC3)no2)=O)C)=O)CN2CCCN1CC2 N1(C(C(C)=C2CC2)=O)CC(C)CN(C(c2cnc3n2CCCC3)=O)C(C)C1 c1(C(N2C(c3ncc(-c4ccc(CC)cc4)o3)CCC2)C)ccc(Cl)cc1 Cc1ccc(-n2cc(C(=O)N(c3ccc4c(c3)CNCC4)C)nn2)c([N+](=O)[O-])c1 Cc1ccc(NC(=O)C(O)C2CN(C(c3n[nH]c4c3COC4)=O)C2)cc1C C1(N=[N+]=[N-])(C(=O)NCCCCC#C)CCN(C(=O)C(C2CCOCC2)F)C1 C(C(N=[N+]=[N-])C(=O)NC1(CNC(=O)C(C)C(=O)OC)CCCC1)OCC N1(C(C2N(C(c3cc(OC)no3)=O)CSC2)=O)CCCC(C(N)=O)C1 N1(C(c2c(CC)cccc2)=O)CCC2(CC1)COC(CNC(=O)COCCO)C2 C1(CNC(C(C)NC(C)=O)=O)CCCN1C(=O)CC1CCCN1C(C)=O C1(CNC(c2c(OC)c[nH]n2)=O)CCCCN1C(=O)C(O)CN(C)C c1(C(=O)OCCC2CCN(C(=O)OC(C)(C)C)C2)cnc(N)c(Br)c1 N1(C(c2c(CC)nn[nH]2)=O)CCCCCC1CC(=O)NC(C)CC(C)(C)OC CC1(C)CCc2c1n[nH]c2C(=O)OCCCOC1CCCCC1 N1(C(c2cc(C)c(=O)n(C)c2)=O)CCN(C(=O)C=CBr)C2CCCCC12 C#Cc1cccc(CC(N2CC(OC)CC2(C)CNC(=O)C#CC2CC2)=O)c1 N1(C(C(c2c(OC)cccc2)OC)=O)CC(C)CN(C(c2cncs2)=O)CC1C c1(C(C)C(=O)N2CCC2CNC(=O)C=CC(F)(F)F)ccn(C)n1 C(c1cscn1)=CC(=O)NC1CC(CNC(C2OCCCO2)=O)C1 C1(OC)CC(N(C(=O)C(c2ccc(C)o2)C)C2CC2)C1(C)C O=C(CCCCC(F)(F)F)N1CCC2CCC(C1)N2C(=O)CCc1cnccn1 N1(C(CCN(CC)CC)=O)CC(NC(c2nc(C)ccc2F)=O)C(C2CC2)C1 c1(C(N(C2CCN(C(=O)C(CCO)C3CC3)CC2)C)=O)cnc2ncccc2c1 c1(C(N2CC(NC(C(C)S(N)(=O)=O)=O)C(O)C2)=O)cc2c(cc1[N+](=O)[O-])OCO2 Cn1ncc(C(N2CCC(CNC(C3(C)CCCCC3)=O)C2)=O)c1C(F)F c1(C(=O)NC2CC(CNC(C3CN(CC)C(=O)N3)=O)C2)cc(Cl)c(F)cc1C C1(C(=O)NC2C(CNC(c3c(C)ncn3O)=O)CCC2)CCc2ccnn2C1 c1(NC(N(CC(=O)NC2CCC(C3CC3)O2)C)=O)ccc(S(=O)(=O)N(C)C)cc1 C(C(C(=O)NC(C1CCCC1)CO)NC(=O)CC1CCCC1O)OC N1(C(C(C)OCC=C)=O)CC2CC(NC(=O)CCCCC(C)C)CC(C2)C1 c1(C(=O)NC2CC(NC(c3c(NC)cnnc3)=O)C2)ccc2c(C)nn(C)c2n1 C1(C(N2CCC(C)(F)CC2)=O)CCCN1NC(=O)Cn1cc(CO)nn1 Cc1ccc(O)c(C(=O)N(C)CC2CCN(C(c3sccc3C(F)F)=O)C2)n1 c1(C(N(C2CN(C(c3c(C(C)C)c[nH]n3)=O)C2)C)=O)cccc2ncccc12 c1(CNC(C2C(CNC(Cc3cc(C)no3)=O)OCC2)=O)cncc(O)c1 NS(=O)(=O)N1CCCC(C(=O)NC23CCCC2CN(C(C2CCCCC2)=O)C3)C1 c1(CN2C(CNC(C(c3ccccc3)C)=O)CCC2)c(I)ccnc1F C(C)(C(C)(C)C)=CC(=O)NCCN(C(c1ccnn1C)=O)CC c1(C(N2C(CC(=O)NCc3ccncc3F)CC(O)C2)=O)cc(F)ccc1F c1(OCC)ccc(C(=O)NC2CCCN(C)C2)cc1[N+](=O)[O-] c1(CCNC(C(C2CC(C)(C)C2)NC(C2(CC)CCC2)=O)=O)nnc(O)o1 C1(NC(C2CCCC2)=O)CC(O)(COCc2ccccc2)C1.C(CO)S c1(C(N(C(CNC(C2(C(=O)NC)CC2)=O)C)C)=O)cc(CO)ccn1 Cc1sccc1C(=O)N(CCCCNC(=O)CC1CC(=O)C1)C c1(NC(C2CCCN2C(=O)C(O)Cc2ccc(O)cc2)=O)c(Cl)cc(Cl)cc1I C(=O)(C(C)(C)C(=O)N(CCNC(=O)C(N1CCSCC1)C)C1CC1)NC c1(C(N2C(CNC(CCc3c(C)n(C)nc3)=O)CC2)=O)[nH]nc([N+](=O)[O-])c1Cl C(CNC(=O)CCSCC(=O)Nc1ccccc1)(CC(C)C)NC(C(C)=CC)=O c1(C(=O)NCC2C(NC(c3c(CCC)occ3)=O)COC2)c(C)ccnc1N c1(C(=O)NCCC2(CNC(C3(CC)CC(C)(C)C3)=O)CC2)cn(C)c(=O)c(C)n1 c1(C(N(C)CC2CCCCN2C(C2CCC2(C)C)=O)=O)ccc2[nH]c(=N)sc2c1 c1(NCCCCCNC(C(C)(C)NC(=O)OC(C)(C)C)=O)cccc(F)c1Cl c1(C(N(C2CCN(C(C(C(C)C)NC=O)=O)C2)C)=O)ccc2c(c1)OCCO2 c1(C(N2CCC(CNC(c3ccc(C)s3)=O)C2(C)C)=O)cccc2scnc12 C1(O)(CC(=O)NCC2C(C)(C)C2)CCN(C(c2cnn(CCCN(C)C)c2)=O)C1 C1(C(=O)NCC2CC23CC3(F)F)CCCC2(CCOCC2)O1 c1(C(c2n(C(C)(C)C)nnn2)NCc2nc(Cl)cs2)cc(O)nc2ccccc12 C(=O)(CC(C)C(=O)NC1CC2(C1)CC(C(=O)N(CC(N)=O)C)C2)OC N1(CC)CCC(C(=O)NCC(C)(CC)NC(c2csc(C(F)F)c2)=O)C1 c1(C(=O)NCC2CC(C)N(C(c3ccoc3)=O)C2)ccc2cnoc2c1 C1(CC(=O)NC2CC(N(C(CCSCCCC)=O)C)C2)COCC(C)(C)O1 C#Cc1ccc(C(=O)NC2(CNC(=O)CCC(=O)CC)CCCC2)cc1F C1(C(N2CC3(CC(CNC(COC(CC)C)=O)C3)C2)=O)OC(C)(C)OC1(C)C N1(C(c2cnc(C(F)F)s2)C(=O)NCCOC)CCC(C)(C)C(COC)C1 c1(C(N2CCN(C(C3(C)C(CC)CCC3)=O)CC2)=O)cnc2cc[nH]c2c1 c1(OC)ccnc(NC(C2CCCN2C(C2CC(F)(CO)C2)=O)C)n1 S(=O)(=O)(CCC(=O)NC1CS(=O)(=O)CC1NC(=O)C1=CCCC1)NC C(=O)(CCCCC(N)=O)NC1C=CCC(C(=O)NCC(CC)(C)C(C)O)C1 C1(C(=O)OC(c2cnnn2C)C)CCc2nnc(Br)n2C1 N1(Cc2nc(-c3ccc(F)cc3)on2)CCc2ccc(Cl)cc21 c1(NC(C)C)ccc(C(=O)N(CC(C)(C)CNC(C2CC2C(C)(F)F)=O)C)cc1 CC(=O)CCCC(=O)NC(CNC(=O)C(C)c1ncco1)C1CCC1 C1(C2(NC(C=C(COC)C)=O)CC2)CCCN1C(=O)CCCC(F)(F)F CC1(C(=O)NCC(O)CNC(c2ccn3ccsc23)=O)CCC(F)(F)C1 CC1(C)CC(CC(N2CC=CCC2)=O)N(C(=O)C#CC2CC2)C1 c1(OC(C)C(N2CC(C)(NC(=O)C(F)(F)CC3CCCO3)C2)=O)ccc(Cl)cc1 N1(C(c2c(C(C)(C)C)ccs2)=O)CCC2CCCN(C(=O)CC3CC3)C2C1 C(=O)(C(C)(CCC)CCC)N1CC(NC(CCC=CC)=O)C(F)CC1 C(=O)(C1CCCn2c(CC)nnc21)NCCC(=C)CNC(=O)CCCCN(C)C CC(C)CC(C(=O)NCC=CCC(=O)NC1CC(O)C12CCC2)N(C)C N1(C(C(CCC)N(C)C)=O)CC(N=[N+]=[N-])CC1C(N1CC2(CC2)C1)=O c1(OC)ccc(C(=O)N(C(C)CN(C(=O)CCCc2cc(C)no2)C)C)cc1 Cc1noc2ncc(C(N3CC4CC3CN4C(=O)C(C)OC3CCCC3)=O)cc12 C1(CC(=O)NC2(CNC(=O)C(O)C3CC3)CCCC2)COCCO1 c1(C(=O)NC(CC)CNC(=O)CCCCN=[N+]=[N-])ccc(S(=O)(=O)N(C)OC)cc1 CC(=O)NNC(=O)C(C)N(CCCC1CNC(=O)C1)C C(C)(CNC(=O)CCSC(F)(F)F)(CC(C)C)NC(c1ncc(C)cn1)=O C(=O)(C(F)(CNC(C1(O)CCC1)=O)C(C)C)NCCCC#C c1(C(=O)NCCC(C)N(C)C(C2CN(C(N)=O)C2)=O)ccnc(C(F)F)c1 C(CN=c1[nH]ccc(=NCC(CO)C2CCC(OC(F)(F)F)C2)[nH]1)c1n(C)cnc1 c1(C(N2C(C(C)NC(c3n(CCC)ncc3)=O)CCC2)=O)cc(C#N)no1 C1(C(N2C(CC(C)C)CC2)=O)CCN(C(=O)COCC(C)(C)C)CC1O C12(CNC(c3c(CCC)occ3)=O)CC(CN1C(C1CC3CC3C1)=O)C2 N#Cc1cncnc1C(=O)NCCOCCNC(c1cccc(=O)o1)=O C(=O)(N(CCC(=O)N(C)CC1CC1C)OC)C1C(=C)CC1 c1(CC)cc2c(CC(=O)NCC3CCC(NC(=O)C(Cl)=CCl)C3)csc2s1 N1(C(C(COC)(C)O)=O)CCCN(CCNC(=O)C(n2nc(C)cc2C)C)CC1 O=C(C1CCSc2ccccc21)NCC12CC3CC1C2C3O CC1CCc2ncc(C(=O)NCC3C4CN(C(=O)CCc5cn[nH]c5)CC34)n2C1 C1(NC(C2(C)C(C)CCC2)=O)CCN(C(c2ccc(O)c(F)c2F)=O)CC1(C)C c1(CN(C(=O)Cc2c[nH]nc2O)C)ccccc1CNC(c1ccoc1)=O Cc1cc(C(=O)NC2(CNC(c3csc4nnsc34)=O)CCOCC2)nc(C)n1 c1(C(=O)NCC(C)(C2CC2)NC(CCOC)=O)ccc(C)c(OC(F)F)c1 CC1COC(C(=O)NCC(C)CN(C)C(c2cnn(Cc3ccccc3)c2)=O)C1 C(=O)(N(CCC(=O)OC)OC)C1C(c2n(CC)ncc2)N(C)C(=O)CC1 c1(C(=O)NCCOCCCN(C(C(CN(CC)CC)F)=O)C)cccc(O)c1F C1(NC(CCN(C)CC)=O)CC2CN(C(C3(C4CC4)CC3)=O)CCN2C1=O c1(C(N(C)CCOCCNC(C2CC2F)=O)=O)ccsc1Br C1(OC)CN(C(=O)COCC2CC2)CCC1NC(c1cccc(O)c1)=O N1(C(Cc2c(C)nc[nH]2)=O)CC2(NC(=O)Cc3ccccc3Cl)CC1C2 Cc1cc(CC(=O)NC2CC2CNC(=O)CN(C)C2CC2)nn1C C1(NC(c2cc(C)on2)=O)CS(=O)(=O)CC1NC(=O)CCOCc1nccn1C C(=O)(CS(=O)C(F)(F)F)N1CC(=C(CNC(C2CN(C)C(=O)C2)=O)F)C1 C(=O)(CCCCC(F)F)N1CCCC(CCNC(C(C)(C)CO)=O)CC1 c1(OCC(=O)OC)ccc(Cl)cc1CNC1CCC1c1cccc(Br)c1 N1(C(C=C(CNC(CCCC#C)=O)C)=O)CCC(CO)C(CO)C1 C1(CC(=O)N(CCNC(=O)CCC2CCCN(C)C2)CC)OCCCC1(C)C C1(N(C(=O)CC(C)(C)O)C)CC2CCC(C1)N2C(=O)CSc1ccccc1 N1(C(CC(=C)C)=O)CCC2CCN(C(c3cc(C)nc(O)n3)=O)CC12 c1(OC)ccccc1C1(C(N2CCOC(CCCO)C2)=O)CCC1 C(C1CCCC1)=C(C(=O)NCCN(C(CC)(C)C)C(c1c[nH]c(C(N)=O)c1)=O)C C1(C(NOCC=C)=O)CC12CCN(C(=O)C(C)(C)CC(F)F)CC2 CCCC(F)(F)C(=O)NC1CC(C(=O)OC)C1(C)C.C1(CCF)C(=O)N1 C(=O)(N=c1cc(COC)n(C)[nH]1)c1cncc(NC(C(CSCC=C)C(C)C)=O)c1 C1(C(=O)NCC(CC=C)NC(=O)CSc2nnnn2CC)CCN(C(C)C)CC1 N1(CCNC(N2CCC(C)(F)C2)=O)C(=O)C2C3C=CC(C3)C2C1=O C(C(CNC(=O)CCOc1ccccc1)C(F)(F)F)NC(C1CCN(C)C1=O)=O CC1(CC(=O)NC2CC(NC(C3(CO)CC3)=O)C2)CCS(=O)(=O)N1 c1(-c2cc(C(=O)NC(C(C)NC(=O)Cc3ccco3)C)no2)ccccc1O CCCC(C(=O)N(C)Cc1ccncc1F)NC(C1C2COCC12)=O c1(OC)c(C(=O)NCC(O)CN(C)C(C2CC(=O)NC2(C)C)=O)c(C)nn1C N1(C(C2CCC(=C)CC2)=O)CC2(COC(CNC(=O)C(n3cc(C)cn3)C)C2)C1 C=CCCC(C)(O)c1nc(-c2ccccc2)nn1C12CC(C(F)F)(C1)C2 N1(Cc2cn(C)nc2)CCC(O)(Cn2nc(-c3ccccc3)oc2=O)C1 N1(C(c2ccc(C#N)o2)=O)Cc2ccc(CNC(C3CC(=C(F)F)C3)=O)cc2C1 c1(CCC)nc(C)c(CN(CC(N2CCN(CC(F)F)CC2)=O)C)s1 N1(C(c2nc(C)nn2C)=O)CCC2(CC1)CN(C(=O)C(=O)NC(C)C)C2C(C)C C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CCC(C)(NC(C2(Cl)CC2(F)F)=O)C1 C(CCCC(C)(C)C(=O)NNC(=O)CNc1cccc(F)c1)NC(C1C(C=C)C1)=O c1(OCC(C)(C)C(=O)NCCCOCC2CC2CC(=O)O)ccc(F)cc1F.CN C12(CNC(C(CCC)(C)C)=O)CN(C(c3cc(C4CC4)on3)=O)CC1CCO2 N1(CC)CC(CNC(C2(COC)CCOCC2)=O)OC(C)C1 N1(C(C=CC(CC)=CC)=O)CC(O)CC1CC.C12CCOCC1NC(=O)C2 n1(CCCSCCN(C(c2ccc(NCC)cc2)=O)C)cc(C#N)c(O)nc1=O N1(C(C23CCC(OC)C2C3)=O)C(C(=O)N(CC(F)(F)Cl)C)C2CC(O)C1C2 C1(CNC(c2ccc(C(C)=O)o2)=O)CC(C)N(C(=O)COC2CCOC2)C1 C1(C(=O)NC2CC(O)CN(C(C3CCSCC3)=O)C2)CC2(CCOCC2)C1 C#Cc1ccc(NC(=O)CC(O)CNC(c2occc2COC)=O)c(C)c1 Cc1cccc(C(N2CC(CCNC(C3CCCN3C(C)C)=O)C(C)C2)=O)c1C C1(CC=C)(NC(C2CCOCC2)=O)CC2CCC(C1)N2C(C1(C)CCCO1)=O Cc1cnc(N2CCCC(NC(C3CCCCN3C(N)=O)=O)C2)nc1C C(=O)(CC1=CCCCC1)NC1CC(NC(C(c2c(OC)cccc2)O)=O)CC1O N1(C(C)=O)CCCC1(C)C(N1CC2CC2(NC(=O)C(C)(C)c2cccnc2)C1)=O CCC(CC)CC(=O)NC(C1CCN(C(C2(CC)CCCC2)=O)CC1)C Cc1cc(C(=O)NCC2CN(C(C3(c4ccncn4)CC3)=O)CCO2)nc(O)c1 Cn1c(C(=O)NC2CCCC2NC(c2ccn3nnnc3c2)=O)ccc1[N+](=O)[O-] N1(C(C2CCC(CNC(c3c(CCC)n[nH]c3)=O)O2)=O)CCC2(CCN(C)C2)C1 c1(C(N(C(C)CNC(c2ccc(SC)s2)=O)CC)=O)ccc(F)c(F)c1N N1(C(CCOCCOCC)=O)CCC(NC(c2ccc(NC(C)=O)cc2)C)CC1 C1(C2CCOCC2)(C(=O)NC2CN(C(C=C(C)C3CC3)=O)CC3C2C3)CC1(F)F N1(C(Cn2c(C)ncc2)=O)CCC(F)(F)C(NCc2cc(I)ccc2Br)C1 c1(OCC(=O)NC(C)CN(C)C(C2CC2c2ccccc2F)=O)cccnc1Cl C(CCC(=O)NCc1ccc(C(=O)NCCCCCSC)o1)=CCC=C Cc1nc(C(N2CCCC(CNC(=O)CN3CCC3C)C2)=O)ccc1[N+](=O)[O-] c1(OC)cnc(C(N2CCC(CCNC(C3(C)CCNC3=O)=O)C2)=O)c(OC)n1 N1(C(C(C)SCCCC)=O)CCN(C(=O)C(c2ccc(F)c(F)c2)C)C(C)C1 C(C(F)(C(=O)N1CCC(COC)C1)C(C)C)NC(c1cncc(OCC)c1)=O c1(C(N2CCC3(C2)CN(C(C2CC4(CC4)CO2)=O)C3)=O)cccc2nncn12 Cc1cccc(C)c1C1(C(=O)NC(C)CCNC(=O)CC2CCCCO2)CC1 N1(C(CN(C(C)C)C)=O)CCCC2(C1)CN(C(C1CCCSC1)=O)CCO2 Cn1ccc2nc(N3CC4CC3CN4c3ncnc4[nH]ccc34)nc(Cl)c12 N1(C(COc2cccc(CC)c2)=O)CCCC(NC(=O)C2=C(C)OCC2)CC1 CC1CN(C(c2cc3ccccc3o2)=O)CCCN1Cc1ccncc1O C1(CNC(c2ccc(CCC)cc2)=O)CN(C(=O)C(C2CCC2)OC)CC1(C)C C1(N(C(=O)C(c2cn(C)nn2)NC(=O)C=Cc2ccsc2)C)CCCC(O)C1 C1(CC(=O)NC(COC)C)CCN1C(c1cn[nH]c1)=O c1(C(N2CCC(NC(COCCC=C)=O)C(F)C2)=O)oc2ccc(F)cc2c1C C(=O)(C1=C(C)CCCC1(C)C)NCC(C1CC1)NC(c1cc(CC)c(F)cc1)=O C1(O)(C(=O)NC2C(C)(C)C(O)C2)CCN(Cc2ccccc2)CC1.C1C2CC3C(C2)C13 C=CCC(C(=C)C)C(=O)N1CCCC(CNC(=O)COC2CCCC2)C1 C(C1CSc2ccccc21)NC(c1cc(CC(C)C)c(N)cc1)=O C12(CC(=O)NC(C(=O)OC)(C)C3CC3)COCC(C1)C2 c1(OC)ncc(C(=O)NC2(C)CCN(C(=O)C(C)c3cncs3)C2)cn1 N1(C(COc2cc(C)on2)=O)CCC2(CCC2)C(NC(C2CC3C=CC2O3)=O)C1 CC1(C)OCCOC1CC(=O)NC1CNCC(F)C1 C(=O)(C(CO)C(C)(C)C)NCC1(COC)CN(C(C2CC3CCC2O3)=O)C1 c1(C(=O)NCCC2(CNC(CN3CC(C)(OC)C3)=O)CC2)cc(C(C)C)nn1C CCC(C)C(O)C(=O)NCC1CC(C(N2CC(C)CCC2CC)=O)C1 C#Cc1ccc(C(=O)NCCCC2(NC(=O)CCSc3n[nH]c(C)n3)CC2)o1 c1(C(CNC(c2c(N)cc(Cl)cc2)=O)NC(C2(O)CC2)=O)cnc2[nH]cnc2c1 c1(N2CC(C(=O)O)CC(CC)C2)ncc2ccc(Br)cc2n1 C1(C(C(C)C)NC(c2cc(C)oc2)=O)CN(C(C2(c3ccno3)CC2)=O)CCO1 c1(C2(C(N3CCC(C(C)O)C3)=O)CCCO2)ccc(Cl)cc1 c1(CN=C(NC2(CO)CC2)NC2CC2)ccc(F)cc1O N1(C(C(COc2cccc(C)c2)C)=O)CCc2c(cnnc2O)C1 c1(C(=O)NCC(C)CN(C(=O)C2=CCS(=O)(=O)C2)C)cc2c(o1)CCCNC2=O S(=O)(=O)(c1c(C)nn(C)c1Cl)NCCNc1c(CC)cccc1 N1(CC(c2c(C)noc2C)(C)C)C2CCC1CN(C(c1cn(C(C)C)cn1)=O)C2 N1(C(C2(F)CCN(C(c3cn(CC=C)nc3)=O)C2)=O)CC(C)OC(C)(C)C1 C1(C(=O)OC)CCOC1NCC1CC(NC(C2CC2c2cncn2C)=O)C1 C(C(CC(C)C)C(=O)NCCc1cc[nH]n1)NC(CCCC)=O C#CCCCC(C)C(=O)N1CC=CC(NC(C2(O)CCCCC2)=O)C1 N1(C(c2cc(C)oc2)=O)CC2CC(C1)N(C(=O)C(C)OCCC(C)C)C2 C(CC(C(=O)NC(C1CCCCC1)CNC(c1n[nH]cc1F)=O)NC(N)=O)SC C1(NC(=O)C=CC=C(Cl)Cl)CC2CC(NC(c3cncc(F)c3Cl)=O)C2C1 N1(C(C2(C=C)CCOCC2)=O)CC(C)N(C(=O)OC(C)(C)C)C(C)C1 C1(CNC(C2(CC=C)CC2)=O)CC(C(=O)N(C)Cc2cccs2)=NO1 C1(CN(C(=O)C(C)(C)CSC)CC)CCN(C(=O)Cc2ccn(C)n2)CC1 c1(C(=O)NC2CN(C(C=Cc3cnc(C)s3)=O)CC2C)cc([N+](=O)[O-])ccc1C C1(C(=O)NC(C(=O)N2CC(N(CC=C)C)C2)CCSC)CC(=O)NC1(C)C C1(C(C(=O)OC)C)CCN(C(=O)N(CCCCC)CCO)C1 C1(C)(CC(=O)N(C)CC2CCCCN2C(C2(CF)CC2)=O)CCS(=O)(=O)N1 c1(OCC=C)ccc(CC(=O)N(CCCNC(c2ncn(C)n2)=O)C2CC2)cc1 c1(C(N2CC(C)(NC(=O)C(CCC)NC(N)=O)C2)=O)c(CC)cnn1C(C)(C)C c1(CCC(N2CC(=C(CNC(C(c3cnn(C)c3)C)=O)F)C2)=O)cccn1C C(=O)(C(C)CC(C)C(C)=O)N(C(CC#CC)CO)C(=O)C1=NOCC1 C(CN(C)N1CCN2C3(CC2C3)C1)N(C)Cc1ccco1.C(C)(C)(C)OC(=O)OC N1(C(c2c(C)coc2)=O)CCCC(C(C)(C)C(=O)NC(C)CCC(F)F)C1 c1(CC(C=C)SN)nnc(-c2ccc(F)cc2)n1-c1cccc(O)c1 N1(C(CC=C)=O)CCOCC(C)(CNC(=O)C(CC)Oc2ccccc2C)C1 C(=O)(C(C)(CSC)NC(=O)C(C)CCOC)NCC(CC)n1cccn1 C1(CNC(c2c(C)nns2)=O)CN(C(C2CCC3CCC(=O)N23)=O)CC12CCC2 C1(CC(N2C(CN(C(c3ccc(O)nc3)=O)CC)CCC2)=O)OCCC1(C)C C1(CNC(CC2(COC)CC2)=O)CCC(C)N(C(c2nn[nH]c2Cl)=O)C1 C1(NC(=O)CCOC2CC2)C(C2CC2)CCN1C(=O)CCOc1ccccn1.CO C1(SCC(=O)NCCCNC(c2cccc(C(C)C)n2)=O)CCS(=O)(=O)C1 CC1CN(C(=O)Cc2ccccc2Cl)CC1NC(c1cnc(=NC)[nH]c1)=O C(=O)(C(C)(C)C(C)(F)F)NC12C(C)OC(C(=O)NCC3COCCN3C(N)=O)(C1)C2 C(CC(C(=O)NOC(C)C)NC(=O)C(F)=C(C)C)=CC c1(C(=O)NC2C(NC(C3C(=C)CC3)=O)COC2)ccc2c(c1)NCCC(=O)N2 C(=O)(C(c1ccccc1)=Cc1ccccc1)NC1C(NC(COCC#C)=O)CC1 c1(C(C)Sc2cc(C3CC3)no2)nc(CC(N2CCC(c3nc[nH]n3)C2)=O)cs1 Cc1ccc(CN(C2CCCC2)Cc2ccccn2)c(O)c1 C1(C(=O)NC(C(=O)NC(C=C)COC)C2(C)CC2)CCCCCC1 c1(NC)snc(C)c1C(=O)NCC1CC(CNC(C2CC3CCC3C2)=O)CO1 c1(C(N2CC(O)(C(C)NC(=O)CC3CCN(C)C3=O)C2)=O)ccc2c(c1)OCO2 C12(C(=O)NCC3(C(N)=O)CN(C(C(C(=O)OC)(C)C)=O)C3)CCC(C)(CC1)OC2 C(CCCCCCC(=O)N1CC(CNC(=O)C(C)(C)C(F)F)C2(CCC2)C1)SC C12(C(=O)NCCCN3CCN(C)CC3)CC(CO1)N(C(c1cnc(O)[nH]1)=O)C2 Cc1cc(NC(=O)C(c2ccc(Cl)cc2)O)cc(C)c1C(=O)O C(=O)(C(CC(C)C)ONC(C1C=CCN1CC)=O)NCCCCC(=O)NC C1(C(C)C)CN(C(c2ccc(CCC(=O)NCCC3(C)N=N3)[nH]2)=O)C1C(C)C C(=O)(C(C(=O)NC1(CNC(=O)C(F)CC(C)C)CCCCC1)C(C)C)OCC N1(C(C=Cc2c(C)ncs2)=O)CCN(C(c2cc(Cl)cn2C)=O)C(CF)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2CCC(C1)N2C(=O)C1=CSCS1 C1(NC(c2c(CC)ncnc2)=O)CCC2(CCCN(C(=O)CCCF)C2)C1 C1(NC(=O)Cc2cncs2)CC2CCC1CC2NC(C1CCc2nc[nH]c2C1)=O c1(C(=O)NCCNC(c2cn(CCC(C)C)nn2)=O)cnc(N(C)C)nc1 c1(NC(C2CC2)C)ccc2nc(O)n(CC3CCOC3)c(=O)c2c1 C1(N(C(=O)CNC(=O)C2CC2)C2CC2)C=CCN(C(=O)Cc2ccc(Br)s2)C1 c1(C(N(C)CCN(C(=O)C(C2CCCCC2)O)C)=O)cc(-c2cc[nH]n2)ccn1 N1(C(C2(CC=C)CC2)=O)CCCN(C(c2ccc(F)c(C(C)=O)c2)=O)C(C)C1 N1(C(C(C(F)(F)F)OC(C)=O)=O)CC(NC(=O)Cn2ccnn2)C(C2CC2)C1 C1(NC(=O)C(F)CC2CCCCC2)CCCCCN(C(c2cncc(F)c2)=O)C1 c1(CN2CC(NC(c3cccc(OC)c3)=O)(CO)C2)ccc(Br)nc1Br c1(C(=O)NCCNC(C2(C)N(C)CCC2)=O)ccc(S(N)(=O)=O)[nH]1 C12(CNC(Cn3c(C)c(Cl)cn3)=O)CCC1CCN2C(=O)COc1cn[nH]c1 c1(CC(=O)NCC(C)N(CC(COC)O)C)nnn(C(C)(C)C)n1 c1(CNC(C2C(NC(C3N(C)CC3)=O)CC2)=O)ncccc1C(F)(F)F Cc1cc(N2CCC3(CCN(C(=O)Cc4cccs4)C3)C2)ncc1[N+](=O)[O-] C(C)(C#CC(=O)NC(c1nnc(O)o1)C)NC(C(C)SCCCC)=O c1(CNC(C2NCC(C(C)=O)C2)=O)sc2ncn(C)c(=O)c2c1C S(=O)(=O)(c1ccc(Br)c(C#N)c1)N(c1ncc(F)cc1O)C Cc1ccc(C(=O)NC2CC(NCc3csc4ccc(Br)cc34)C2)c([N+](=O)[O-])c1 CC(C)S(=O)(=O)CCC(N)C(=O)Nc1cc(Br)cc(C(C)(C)C)c1O C1(NC(COCC(C)(C)C)=O)CC1C1CCN(C(C2(CF)CC2)=O)CC1 C1(C(N(C)CC2CCCN2C)=O)CC(F)(F)CN1C(C1CCCC1)=O c1(C(=O)NC2(C)CC(NC(c3ncoc3C3CC3)=O)C2)cncc2c1CCC2 c1(C(C)=O)ccc(C(=O)N(CCCCCNC(=O)Cn2ccc(C)n2)C)s1 C#CC1(O)CC(C(=O)NCCC2CN(C(=O)Cc3cccc(CC)c3)CCO2)C1 C1(C#N)(C(N2CC(C(C)NC(c3ocnc3C3CC3)=O)C2)=O)CCS(=O)(=O)CC1 c1(C(=O)NC(C2CCCN2C(=O)C=C(C)C(C)(C)C)C)ccc2[nH]ccc2c1 C1(C(N2CCCC(N(C)C(C3CCCCC3)=O)CC2)=O)CCCC2(CCC2)O1 CCC(C)CCCC(=O)NCC1CC1CC(=O)NCC(C)C(C)CC C1(CNC(=O)CN2CCCC2)CCCN(CCCn2[nH]c(C3CC3)nc2=O)C1 c1(CNC(C2C(NC(c3ccc(C(F)F)cc3)=O)C2)=O)ccc(F)nc1F c1(CC)cccc(C)c1NC(=O)CNC(=O)CC1C=CCCC1 C1(C(=O)NC(CC#C)C(=O)NCc2ncc(C)cc2C)CC(=O)CC12CCC2 C1(C(N(C)Cc2cccc(CNC(=O)Cc3ccco3)c2)=O)CC(=O)OC1(C)C CC(CCC(=O)N(C)CCC1CCC1)NC(=O)C(C)(C)O CCCC(C)(C)CC(=O)N1CCCCC(C(=O)NC2CCCC2(C)C)C1 C1(NC(C(CO)OC)=O)CC12CCN(C(c1cnn3c1NCCC3)=O)CC2 n1(CC)ncc(C)c1C(=O)NCCCC(C)(C)NC(=O)C(C)C1CCOC1 N1(C(c2ccc(-c3cccc(Cl)c3)s2)=O)CC2CN(Cc3ccc(F)cn3)C2C1 C1(NC(C2(CC(C)C)CC2)=O)C=CC(C)(C)CC1.C1CC(=O)NCCCCCO1 c1(NC(C)=O)cc(CNC(=O)Nc2cc(-c3ccccc3)cn2C)oc1C N1(C(c2scc(C)c2)=O)CCOC2CN(C(=O)CC(C(C)C)C(C)C)CC12 c1(C(=O)OC)nc(=NCCc2ccc(C(=O)O)cc2Br)c(Cl)c[nH]1 c1(C(=O)NC2CCC(C)(CNC(CCN(CCC)C)=O)C2)nc(C)c(C)nc1C c1(COC(C=C(C)Cl)=O)ccc(CC(F)(F)F)nc1 Cc1ncc2n1CCC(c1nc(C3CCCO3)nn1CCS(N)(=O)=O)C2 C12(C(=O)NC(CN(C(c3ccc(C(=O)OC)nc3)=O)C)C)CCCC(C1)C(=O)N2 S(=O)(=O)(c1sc2ccccc2c1C)N1CC2(CCC(C(=O)OC)O2)C1 N1(C(C2(C)CC=CCC2)=O)CCCC2(CCN(C(C3CCNC3=O)=O)C2)C1 C1(CNC(C(C)=C2CCC2)=O)CN(C(c2cc3ccsc3[nH]2)=O)CCC12CCC2 Cc1oc(CO)cc1C(=O)NC(C1CCCC1)CNC(c1ccc(N)cc1)=O N1(C(C(C)OC)=O)CCC(C2CC2NC(c2ccc(F)c3c2OCC3)=O)CC1 C1(C2CCCN(C(c3nnsc3C)=O)C2)(NC(C2C(CC)C2)=O)CC1 C1(C(=O)NC2C3CC(NC(c4c(Cl)cn(C)n4)=O)CC32)CCn2ncnc2C1 Cn1nc(C(N2CC3(C2)CN(C(=O)C(O)C(F)(F)F)C3)=O)c2ccsc12 N1(C(c2cc(C)[nH]c2C)=O)CCCC(C)(C)C1C(N1CC2(CNC(=O)C2)C1)=O C1(OC)CSCCN(C(=O)Nc2ccc(Cl)cc2O)C1 C1(F)(C(=O)NCCCN(C(c2ccc(C)s2)=O)CCO)CC2(CCC2)C1 c1(NC(C2CC3CC2CN(C(C2(Cl)CCC2)=O)C3)=O)cncc([N+](=O)[O-])c1 c1(OC)cccc(-n2nnnc2C(c2cc(C)sc2C)NCCC(O)C2CC2)c1 N1(C(C2CCCN(C(Cc3n(C)ccn3)=O)CC2)=O)CC2CCCC(O)C2C1 Cn1cc(CC(=O)NC2(CNC(C3CC(F)C3)=O)CC2)cn1 C1(O)(Cn2cc(CC(C)(C)O)nn2)CCN(C(=O)Cc2cncn2C2CC2)C1 O=C(CCC1C(=O)Nc2ccccc21)NC1CN(C(c2cccnc2)=O)CC1F CC1(NC(c2cccc(CC#N)c2)=O)CCN(C(c2csc(O)n2)=O)C1 C(CC(=O)NCCCc1ccco1)N(CC=C)C(C1CC1c1ccco1)=O C(=O)(C1CCCc2nc[nH]c21)N1CC(CC(C)NC(c2ncn(C(C)C)n2)=O)C1 C1(OC)CCC(N(C(C2(C)CC3(CC3)C2)=O)C(c2cc(CC3CC3)c[nH]2)=O)CC1 c1(C(N2CCC(O)(CN(C(CSCC=C)=O)C)C2)=O)ccn2nnnc2c1 C(=O)(CCCC(C)C)NCC1CCCN(C(Cc2c(C)nc(C3CCC3)s2)=O)C1 N1(C(CCOCCC)=O)CC2CC(C1)N(C(C1CC13CCSCC3)=O)C2 CC#CCCCC(C)(c1nnnn1C)Nc1ccc(OCC23CC(C)(C2)C3)c(F)c1 CCCC(CCC)C(=O)NCC1(NC(=O)CN2CCCNC2=O)CCC1 C1(NC(c2c(CC)nc[nH]2)=O)(COC)CCN(C(c2nn(C)cc2Br)=O)CC1 C1(OC)CC(CNC(=O)CN2CCOC2=O)N(C(=O)CCC2(C)CCC(=O)N2)C1 c1(C(=O)NC2CCCC2OCCOC)ccc2c(c1)CCCC2NC(=O)CSC CC1OC2(C(=O)N(C)CCN(C(=O)CCOc3cccnc3)C)CC1C2 O=C(C(Cn1cccn1)NC(C1CC12CCC2)=O)NCc1nncs1 c1(C(N(CC(CNC(CC(CC)C2CC2)=O)(C)C)C)=O)ccc(Cl)cc1C(F)F Cc1cc(C(=O)NCC(C)(CO)NC(C2(C3CCCO3)CC2)=O)cc(F)c1 C1(OC)CC(CNC(=O)CC23CCC(CC2)C3)N(C(=O)CSCC(N)=O)C1 N1(C(CCCC(C)=O)=O)CC2OCCN(C(=O)C3Cc4ccccc43)C2C1 c1(C(N2CC(N(C(C(C)n3ccnn3)=O)C)C2)=O)ccc(Cl)c2ccccc12 C(=O)(CCCCC(C)(C)C)NCC(CCOC)NC(=O)CCC(=O)c1cccs1 c1(C(=O)NC2CC(OC)CN(C(c3cnn[nH]3)=O)C2)cc2cccc(O)c2[nH]1 Cc1ncnc(N(C(c2ccc(Br)cc2F)=O)CC2(O)CNC2)c1Br CCC(C(=O)NC(C)CNC(=O)CCC1CCOC1)SC C1(CC)CN(C(=O)CC2CCCCC2NC(=O)CSCC(N)=O)CCS1 C(C(C(=O)N1CC(c2ccccc2)C1)C(C)C)NC(CC1(CC)CCC1)=O CC1CCN(C(=O)CC2CN3CCC2CC3)CC1NC(=O)C=Cc1cncn1C Nc1ncc(Br)nc1C(=O)NCC#CCNC(c1ccccc1C1CC1)=O Cc1c(Br)c(CCNC(N2CCOC(c3ccccc3)C2)=O)nn1C CCCC(CC(=O)NCCC1(C)CCCC1)NC(c1cc(C(C)=O)[nH]n1)=O C(C(F)(C(=O)NCCC1(C)CC1)C(C)C)NC(CC1CCC(C)CO1)=O C1(C(N2CC(CNC(CC(=O)OCC)=O)C(C)CC2)=O)CC2(CCOCC2)C1 C=C(Cl)CCC(=O)N1CCCC1C1(NC(c2cnoc2C)=O)CC1 C1(c2nnnn2-c2ccccc2Cl)(NCc2ncc(SC)cn2)CC2(CCC2)C1OC Cc1cc(C#N)ccc1C(=O)NC1(C(=O)Nc2ccc3ccoc3c2)CC1(C)C C(=O)(CCC(=O)NCC1(O)CC(C(=O)NCC(C)=C(C)C)C1)NCCC C(C(CC(C)C)C(=O)N(C)C[Si](C)(C)C)NC(C1(CC)CCCCO1)=O C(CC(O)CC(=O)N(C(C)CNC(c1n[nH]c(C)c1Br)=O)C)SC c1(OCC)ccc(C(N2CCCCC(CNC(=O)CCC(C)SC)C2)=O)cc1Cl C=CCC(C(=O)NC1(C)CCC(=O)N1)NC(=O)CC(=O)OCC C#Cc1cccc(C(N2CCC3(CC2)CC3NC(=O)C(C)CC2CC2)=O)c1Cl C(C)(CCCCNC(=O)C(C)NS(C)(=O)=O)NC(c1ccc(COC)s1)=O N1(C(Cc2ccc(C)s2)=O)CCN(C(c2coc3c2COC3)=O)C(C)C1C n1(CCCOCC)c(N2CCOC(c3cc(C)no3)C2)nnc1-c1cc(I)cs1 C1(C(N(CCCF)CC)=O)CN(C(=O)CC2CCCCC2)CC1OC.CCS C1(C#N)(CNC(C2(CNC(c3c(C)n(C)cn3)=O)CC23CCC3)=O)CCOCC1 C(CC(C)C(=O)N1CCCC1C=CC(=O)NCC(=O)N(C)C1CC1)=CCC c1(C(=O)NC2C(NC(c3ncoc3C3CC3)=O)CCC2)cc2occ(Br)c2[nH]1 N1(C(c2c(CC)nc(C)o2)=O)CCC2(CCCCC2NC(c2conc2C)=O)C1 c1(CNC(COCC(=O)NC)=O)nnn(C)c1C(=O)NCC1CC2CCC1C2 c1(CC)nc(C)[nH]c1C(N1CCCC1C(C)NC(=O)C=CC(C)(C)C)=O C1(OC)CC(CNC(c2cc(C)n(C(CC)CC)n2)=O)N(C(=O)CNC(N)=O)C1 Cc1cc(C(=O)NCC2CC(C)N(C(=O)CCS(C)=O)C2)ncc1C#N CCC(C)CCCC(=O)N1CCC2(C1)CN(c1nccc(COC)n1)C2 c1(-c2c(OC)ccc(F)c2)cc(C(N2CCCOCC2)=O)cc2c[nH]nc12 CC(C)(C(=O)NC1CCC(C)(CNC(=O)CCC2(C)CCC(=O)N2)CC1)C(N)=O N1(C(C2C(C)C2C)=O)CCCC(C2CC2NC(C2CCOCC2)=O)C1 C12(CNC(CC(C=C)C)=O)CCCC1CN(C(c1[nH]ccc1C1CC1)=O)C2 C(CC(F)F)(C(=O)N(CC(C)C#N)C)N(C(c1c(CC)c[nH]c1)=O)C c1(OC)cc(C(=O)NCC2CC2NC(c2cnoc2C)=O)cc2c(C)c(C)[nH]c12 N1(C(c2c(C)cnn2C)=O)CCC(NC(=O)CC2C=CS(=O)(=O)C2)C(C(N)=O)C1 c1(C(=O)NCC(CNC(C(CC#C)C2CC2)=O)(C)O)cnc(O)c2ccccc12 CC1CN(C(=O)COCCOCCO)CCN1C(=O)C1=CCCCC1 c1(C(=O)NC2(CNC(c3nn(CC)c(=O)cc3)=O)CC2)ccc2ncccc2c1 c1(CS(N2C(C)(c3cn(C)nn3)CCC2)(=O)=O)ccccc1N=[N+]=[N-] c1(C(=O)NCCC2(O)CNC2)ccc(O)cc1.CCC(C=O)Sc1ccccc1 CC(C(=O)NC1(C(=O)NCCOCC(C)(C)O)CCN(C)C1)S(N)(=O)=O C12(C(=O)NC3CCC(N(C(CC4N(C)CCC4)=O)C)CC3)CCCC1CCC2 C12(NC(c3c(CC)nc(C)o3)=O)CCCN(C(c3cc(C(N)=O)c[nH]3)=O)CC1C2 C1(CN(C)C)CCCN(C(N(C(C)(C)C)CC)=O)C1.C(C(C)C)OCCOC(=O)O CC1CCCCC1(CNC(c1cccc(F)c1Cl)=O)NC(C1(N=[N+]=[N-])CC1)=O N1(C(C2(CC(C)C)CC2)=O)CCC(O)(CNC(=O)C(C)(C)N(C)C)C1 C1(C)(CNC(C2CC(C)OC2)=O)CCCN(C(=O)CCNC(=O)CO)C1 N1(c2n(CC=C=C)nnn2)CCN(C(C)CC)CC1 Cn1ccc(C(=O)NCC2(C)CCN(C(=O)CCCc3cccs3)C2)c1C1CC1 C=CC(CC)CC(=O)N1CC2CC(CNC(=O)Cc3nc(C)c(C)s3)C2C1 N1(C(C2(CCC=C)CC2)=O)CCC(NC(C2CCN2CC)=O)C12CC2 c1(C(=O)NCCN(C(C(C2CCC2)OC)=O)CC(C)O)cc(O)cc(F)c1F c1(C(N(CCNC(c2cn(C(C)C)cc2C)=O)CC)=O)cnn2ccncc12 N1(C(Cc2c(C)noc2)=O)CCCOC(CNC(c2nc(O)c(C)s2)=O)C1 c1(CC(C)C)ccc(CC2(CNC(=O)OC(C)(C)C)CC(C(=O)O)C2)o1 c1(C(N(C(C)CNC(C2CCCC2C(F)F)=O)C)=O)n[nH]c2c1CCCCC2 c1(CC)cc(C(=O)N(CC(C)NC(c2cc(CO)n(C)n2)=O)C)oc1CC c1(C(=O)Nc2n(C)nc(C3CCC3)n2)ccnc(O)c1Br c1(C2CCN(CC3CCC(=O)O3)CC2)cccc2cc[nH]c12 c1(OC)cc(Cl)ccc1C(N1CC2C(N(C)C(c3ccc(Cl)o3)=O)C2C1)=O N1(C(Cc2c(C)n[nH]c2)=O)CC(C)C(C)(CNC(=O)Cc2c(Cl)cnn2C)C1 N#Cc1ccnc(N2CCN(CCCNCC3CC4CCC3C4)CC2)c1 C1(C)(CCC(=O)NCC=C(C)C)CN(C(=O)CN2CCCC2)C1 c1(C(=O)NC2CCC(C)(CNC(CC(=O)OCC)=O)C2)ccn2ncc(C)c2n1 C1(CC(=O)N(CCCC(=O)N(C2CSC2)C)C)CC(C2CC2)C1 c1(OC)ccc(CC(=O)NCC(C2CC2)NC(C2COCCO2)=O)c(Cl)c1 CCC(CC(=O)N1CC(O)(CNC(=O)CC(F)(F)C(F)(F)F)C1)C(C)(C)C c1(CNC(c2c(CNC(C(C3CC3)SC)=O)c[nH]n2)=O)ccccc1F CC(C(=O)N1CC(CC(F)(F)F)C1)n1ccnc1 c12cc(ccc1Cl)CC(=O)N1CCN(CC1CO)C2=O.C1(OC)CCCC1CF C(=O)(C(F)C(F)(F)F)NC(CCN(C(c1c(C)oc(C(C)(C)C)n1)=O)C)C(C)C CC(C(=O)N1CCN(C(c2cccnc2C(F)F)=O)CC1CCO)C(C)(C)C Cc1ccc(C(n2cc(CCNC(=O)CCc3nccs3)nn2)C)cc1 C1(CC(=O)N(CC2CCC2)CC2CC2)CCCCC12CC2 CC1(C)Cc2[nH]nc(C(N3CC4(CCN4C(C4CC4C4CCCC4)=O)C3)=O)c2C1 CCCC(O)CN(C)C(C1(CCNC(=O)C(COC)OC)CCC1)=O CN1CCCCC(NC(=O)C#CCNC(C2CC(C)(C)CCO2)=O)C1=O C(=O)(C1COc2ccc(Cl)cc21)NCCCN(c1nnc(C#N)s1)C C1(CCOC)(NC(c2sccc2F)=O)CCN(C(C2CC(=C(F)F)C2)=O)C1 C(CNC(=O)CN(C(=O)C(C)CSC)CCOC)(C(C)C)OC C(=O)(C#CC1CCCOC1)NC1CCN(C(c2cc(OC)c(N)cc2)=O)CC1F c1(CN(CC(=O)NCC2C(CNC(C3(C(C)C)CCC3)=O)C2)C)ccc(Cl)cc1 Cc1cccc(N2CCC(C(=O)NCCN(C(=O)C(O)C3CC3)C)C2=O)c1 CCC(C)(O)C(=O)NCC1CCCCN1C(c1csc(Br)c1Cl)=O S(=O)(=O)(c1ccc(Cl)c(F)c1Cl)NC1CN(C(=O)OC(C)(C)C)C1 c1(C(=O)NCCC(C)(C)N(C(=O)C(C(C)O)N(C)C)C)cc(=O)n(C)cn1 Nc1cc(Cl)cc(Cl)c1C(=O)NC1CC(NC(c2noc3c2CCCC3)=O)C1 c1(N2CC=C(C)CC2)ncnc(NC(C)Cc2ncn(C)n2)c1C c1(C(C)(C)NCC(C)Sc2ccccc2)ccccc1C#N c1(COc2ccc(CNC(NCC=CC)=NC)cc2)ccc2c(c1)OC(C)(C)O2 C(N=c1[nH]c(=NC2CC(C#N)C2)c2ccccc2[nH]1)C1OCC(CC#N)C1 C1(CNC(CSCCC)=O)C(C)CCN1C(=O)C(C)CN1CCCCC1 N1(C(CC(C)n2ccnc2)=O)CCOC(C(C)(C)C)C1 Cc1onc(CO)c1C(=O)NCC(c1ccccc1)NC(=O)COc1ccsn1 C(C)(C)(CCC(=O)N1CCOCCC1C(=O)NC(C)CC1CCC1)OC c1(C(=O)NCC2N(C(CCC)=O)CCOC2)cnc2ncccn12 Cn1cccc1CNC(=O)C(CO)NC(=O)CN=[N+]=[N-] c1(NC(C2C(NS(CCCC)(=O)=O)CCCC2)=O)c(OC)ncnc1Cl Cn1cc(C(=O)NOc2nc[nH]n2)cn1.C1(Cc2ccoc2)C(=O)N1 c1(N(C2CNCC(C)C2)Cc2cc(C)nn2C)ccn2ncc(C#N)c2n1 C1(NC(N(C)Cc2c(C)n(C)nc2)=O)CCc2nc(N3CCN(C)CC3)sc2C1 c1(CC(=O)N(CCC)CCNC(c2cc[n+]([O-])cc2)=O)ccc(C)c(F)c1F Cc1cnc2nccc(N3CCC4(CCC(CC(=O)N(C)C)C4)C3)c2c1 c1(C(N(C)CC2(NC(=O)CC3CCCC(=O)N3)CC2)=O)cc2ccccn2n1 CCC(C)(C)C(C)CC(=O)NCCC1(O)CN(C(=O)Cn2ncc(Br)n2)C1 c1(C(=O)NC2CC(CCNC(C3C4C5CCC(C5)C34)=O)C2)ccc2ccoc2c1 Cc1cc(Cl)cc(C)c1C(=O)NC1CCCCC1NC(C1(CO)CCOC1)=O N1(C(c2c(C)c[nH]c2)=O)CC(NC(C2CCCN2C(=O)CC(C)(C)C)=O)C2(CC2)C1 C1(CNc2cc(F)c(-c3cccc(OC)c3)c(F)c2)CCC2C(CC1)C2(F)F c1(C(N2CCC(F)(C(=O)Nc3c(COC)cccc3)C2)=O)cccnc1NC C1(CC(=O)NC2C(C)N(C(c3ccc(N(C)C)nc3)=O)CC2)CCCC(C)(C)C1 c1(OC)c(Br)cc(Br)c(C(=O)O)c1C.c12cccc(c1)C(=O)N2.C1(=O)CO1 C(=O)(CC(C)(C)C(F)F)N(CCC(C)NC(C1(OC)CCOC1)=O)C C1(OC(C)=O)CN(C(=O)OC(C)(C)C)CCC1F.C12CCCN(C1)C2 c1(C(C(=O)OC)OC2CNC2)ccc(Cl)cc1F C(N=c1[nH]c(N2CC(C)OC(C)C2)nc2cccnc12)c1ccc(CC)cc1 N1(C(C(c2ccccc2F)C)=O)CC2=C(C1)CN(C(=O)Cc1csnn1)C2 C(=O)(C(F)(F)CCc1ccccc1)NCC(CN(C(C(C)=C1CC1)=O)C)(C)C n1(CC)c(C)nn(CC(=O)NC2CCC(NC(c3ccc(C)s3)=O)CC2)c1=O C1(NC(C2(CCCC)CC2)=O)CN(C(c2cnncc2OC)=O)CC1C c1(OC)cc(C(=O)NCC2CC(NC(=O)CC3CCCS(=O)(=O)C3)C2)cc(F)c1 c1(C(N2CCCC(NC(CCCC(CC)C)=O)C2C)=O)cccc(S(C)(=O)=O)c1F C1(C(N(C(CC)CC)C)=O)CCN(C(=O)C(C)CC(F)(F)F)O1 CC1OC(=O)NC1C(=O)NCCC1(C)CCN(C(=O)C=C2CCCCC2)C1 c1(C(=O)NCC2(C)CCC(NC(C=C(CC)CC)=O)C2)cc2ccccc2[nH]1 N1(C(c2c(CC)cccn2)=O)CCCC(NC(C2(F)CCCC=C2F)=O)CC1 C(C(=O)N1CCC(C(=O)OC)O1)(c1ccnn1C)NC(COCC=C)=O N1(C(C2(CC)CN(C(C3CCCCO3)=O)C2)=O)CC(C)(C)C1C(C)C N1(C(C2(C)CCCC2)=O)CC2CCC1C1CN(C(C3CCC3(F)F)=O)CC21 C(=O)(CCC(=O)N1CCC(C)C1CNC(=O)C=CCO)OC n1(CC)cnc2c(N3CCCC(CF)C3)nc(=NCc3ncc[nH]c3=O)[nH]c12 c1(NC(c2cccc(N)n2)=O)c(Cl)cc(F)cc1Cl c1(CCC=C)ccc(C(=O)NCCC2(O)CN(C(C3CC(CF)C3)=O)C2)cc1 Cc1cc(Cl)nc(CNC(=O)NCC(c2cccc(Br)c2)C)c1Br N1(C(C(OC)OC)=O)CC(CC(=O)NCc2ccc(C(N)=O)nc2)C2(CC2)C1 S(=O)(=O)(c1cccc(=NCCCCCO)[nH]1)NC(COCC)C(C)C C1(CCNC(=O)COCC(F)(F)F)CCN(C(=O)CC2CC(C(F)F)C2)CC1 Cc1cc2occ(CC(=O)NC3CCN(c4cc(N(C)C)ncn4)C3)c2cc1C CCC(C)(CO)C(=O)N1CC2(CNC(c3coc(CC4CC4)n3)=O)CCC1C2 CC(C)CCCC(C)NC(C1CC(F)CN1C(=O)CC(C)C(F)F)=O CCCS(=O)(=O)c1ccc(C(=O)NCC(C)NC(=O)CCCC(C)(C)C)cc1 C1(CNC(C2CCNC2=O)=O)CCCN1c1ccncn1 C1(CN(C(=O)Cc2cccc(OC)c2)CC)CN(C(=O)CC2CSC2)CCO1 C1(NC(c2c(CC)csc2)=O)CCCCC1NC(=O)C(C)(C)N1CCOCC1 Cc1nnc(=NCC2CCCC(NC(C3CC4CCCC(C3)C4)=O)C2)[nH]c1C N1(C(c2c(C)nc(C3CC3)s2)=O)CC(O)(C2(CNC(C3(C)COC3)=O)CC2)C1 C1(CNC(CN(C)C(c2cccs2)=O)=O)C2CN(C(=O)CSCC(N)=O)CC12 C1(C(=O)NCC2C(NC(COC(C)=O)=O)C2)CC(=O)N(C)C1c1ccccc1 CN1CC=C(C(=O)NCC2CCC(C(=O)NC3CCCC3(C)N(C)C)CC2)C1 CN(C(=NCc1ccc(Cl)nc1)NC1CCC1)Cc1ccc(F)cc1Br c1(OC)ccnc(F)c1C(=O)NC(C)CNC(c1n[nH]c(C)c1F)=O Cc1cc(NC(=O)CC2CC(NC(c3ccc(C(N)=O)o3)=O)C2(C)C)cnc1O C12(C(N)C(N3CCC(c4cccc(OC(F)F)c4)C3)=O)CC3CC(CC(C3)C1)C2 Cc1nc(C)c(C(=O)NC2COC3(C2)CN(C(C2CCCC2(F)F)=O)C3)c(C)n1 C1(NC(c2c(Cl)c(C)n(C)n2)=O)CCCCN(C(=O)CC23CCC(C)(C2)OC3)C1 CCCC(C#N)C(=O)NCc1ccc(CN(C(=O)C(O)C(C)C)C)cc1 C1(C2CCCCC2)(C(N2CCC(F)(CNC(CC(C)F)=O)C2)=O)CC1 C(CC(C)(C)C)(C(=O)NCC1(OC)CCN(C(=O)CC2CC3CC3C2)C1)OC C1(C(=O)Nc2cccc(-c3noc(C4CC4)n3)c2)CC2(CCC2=O)C1 c1(CC)nc(C(N2CC(CNC(c3nc(C(C)(C)C)no3)=O)CC2C)=O)c(N)s1 CCC(C)(C(=O)N1CC2(CC(NC(=O)CN3CCCCC3)CO2)C1)C(N)=O C1(C(=O)OC)CC(n2cc(CN)nn2)CN1C(C1(C(F)F)CCCO1)=O C1(NC(c2c(C)noc2N)=O)CCCN(C(C2CCN(C)CC2)=O)CC1 c1(NC(c2cc(CC)on2)C)ccc(S(=O)(=O)NCCc2nc(C)no2)cc1Cl N1(C(=O)N(C)C)CC(O)CC1C1CC1.c12ccoc1NC(=O)C2C c1(C(=O)NC2CC2C(N2CCC(N3CCOCC3)CC2)=O)cc(Cl)cc(Br)c1F c1(CC(=O)NC(c2cccc(Cl)c2)CNC(C2(CC)CCC2)=O)nn(C)cc1Cl n1(CCC(=O)NCCN(C(C2CN(C(C)C)C(=O)C2)=O)C)cnc([N+](=O)[O-])n1 n1(CCC)ccc2cc(NC(c3cnn(CCC(=O)OCCO)c3)=O)ccc12 C(=O)(C#CC1CCC1)N(C(C(C)C)(C)CNC(C1CN(C2CCOCC2)C1)=O)CC Cc1c(NC(C)C)cccc1C(=O)NCCN(C(=O)CCc1cn(C)nn1)C N1(C(C2C3N(C(C4OCCC(C)(C)C4)=O)C(CC3)C2)=O)CC(C2CC2(F)F)C1 c1(CC)c(C(N2CC(CC(C)NC(C3(C)CC4CC4C3)=O)C2)=O)csc1C N1(C(c2c(CC)cco2)=O)CCN(C(c2cocn2)=O)C(c2cccc(F)c2)C1 N(C(=NCCSc1ncc(N(C)C)cn1)NCCF)CC1C(C)CCCC1 Cc1oc(C(C)C)nc1CNCC=CCNC(C1C(NC(=O)C(C)C(C)C)C1)=O C(=O)(C(CCS(C)=O)N(C)C)NCCOCCCNC(CCc1ncc(C)[nH]1)=O C1(F)(CNC(C2C(NC(C3CCCC34CC4)=O)CCC2)=O)CCOCC1 C1(C(N(C(CC#C)C)C)=O)CN(C(c2sc(C)cc2C)=O)CC1OC C1(C(=O)NCC(C2CCOC2)OC)CCCC1NC(=O)C(C1CCCCC1)C N1(C(COCC)=O)CCC(NC(c2cnc(C(F)F)cc2C)=O)C(O)C1 C(C(C)(C)CNC(=O)Cc1ccco1)N(C)C(c1nc(Br)c[nH]1)=O c1(C(=O)OCc2c(C)ccs2)ccc([N+](=O)[O-])c(N)n1 N1(C(Cc2cc(OC)c(O)cc2F)=O)C2CCCC1CN(C(C1(F)CC1C)=O)C2 c1(SCCN(C)CCNC(=O)NCCC2CC2)ccc(Br)cc1 c1(C(=O)NC2(COC)CN(C(C3C(=C)C3)=O)C2)cccc(OCCC)c1 C(=O)(C(F)(F)N(C)C)NCCCN(C(=O)CCCc1ccccc1)C C(=O)(C1=CCCC1)NCCC(CNC(C1C(c2ccccc2)C1(C)C)=O)OC c1(C(=O)NCC2CC(CC(C)(C)C)C2)ncc(Cl)cc1Cl c1(N2CCC(C)S(=O)CC2)nc2c(c(=NC3CCN(C)C3)[nH]1)SCC2 C1(NC(CCCOCCC)=O)CCCC(C(=O)Nc2cc(N)ccc2C)CC1 CCCC(CC)C(=O)N(C)CCOCCC(=O)N(C)CCC1CCCO1 C1(C(=O)NCC2CN(C(C3CN(CC(F)(F)F)C3)=O)C2)CC2(C1)CC1(CCC1)C2 N1(C(C)C)CCN2C(=O)C(NC(c3ccn4cnnc4c3)=O)CC2C1 CN1CC(O)CC1C(=O)NCCC(O)CNC(c1ccc(C2(C)CC2)cc1)=O N1(C(CC(COC)C)=O)C2CCC1C(F)C(NC(=O)C1=CCOCC1)C2 c1(C(N2CC(C)C(NC(c3cnc(O)c(Cl)c3)=O)C2)=O)csc(S(N)(=O)=O)c1 CCCCCC(C)CC(=O)NCC1CN(C(c2cc(C)cnc2N)=O)CC12CC2 c1(C(N2C(CO)CC(NC(c3nccc(C)c3)=O)C2)=O)nccc(C#N)c1F c1(C(=O)NCC2C(NC(c3ccn(CC)n3)=O)C2)cccc(OC)n1 C1(CC(=O)NCC(COCC)C)CC(O)CN1C(c1cc(CC)c[nH]1)=O C(=O)(CC(CCCC)NC(=O)CN1CCCCC1)N(C1CC1c1ccco1)CC#C Cc1cc(C(=O)NC(C)C(CO)NC(=O)COCC(F)F)ncn1 CCCCCC(=O)NCC(=O)NC1(CNC(C2CCC(=O)N2)=O)CC(OC)C1 Nc1cc(Cl)c(Cl)cc1C(N1CCN(C(C23CCCC2C3(F)F)=O)CC(O)C1)=O c1(C(N2CC(C)C(NC(c3cncc(Br)c3)=O)C2)=O)ccc(Cl)cc1F C(=O)(C(C)C(C)COC)NCC1C2CN(C(c3n(CC)ncn3)=O)CC21 C(=O)(CCCC(C)(C)C#N)N1CC(CNC(C(C)C(F)(F)F)=O)N(C)CC1 C12(F)CCCN(C1)C2=O.C=C(Cl)CCC(=O)NCCOc1ccncc1 CN1C2CCCC1CC(N(CCO)CCOc1ccc(-c3nn[nH]n3)cc1)C2 N1(C(C=CC(C)C)=O)CC2COCC(C1)C2NC(C1COC2COCC12)=O C(=O)(C(C)(O)C(F)(F)F)NC1CC2(CC(CNC(c3cccc(C#C)c3)=O)C2)C1 C1(CNC(C2N(CC)CCOC2)=O)CN(C(C2CCCC(F)C2)=O)CCN1C C(=O)(CC1OCc2ccccc21)NCCCNC(c1cnc(C)nc1C(C)C)=O CCCC(CCC)CC(=O)NCC1CC2CCC1N2C(c1cccn(O)c1=O)=O C1(C)(CNC(C=CCOCCOC)=O)CCN(C(=O)C(C)N2CCC2)C1 N1(C(C2CC(OC)C2)=O)CC(NC(c2nccn2C(C)C)=O)CC12CCC2 c1(OC)c(C(=O)N(C2CCCN(C(=O)C=C(C)C)C2)C)cccc1F C(C1CCOc2ccccc21)NC(=NCCCF)NCCCN1CCCCC1 c1(C(=O)OCC)ccoc1C(=O)NCC(C)N(C)C(c1ccnn1C1CCC1)=O N1(C(CCCN(C)C)=O)CCC(C(=O)NC2CC2c2ccccc2)C12CC2 C1(NC(CC2CCC(C)C2)=O)CCN(C(C2CCCC2)=O)CC1(C)C c1(C(N2CC(NC(C3(F)CCCC3)=O)C(F)C2)=O)ccc2nc(C3CC3)cn2c1 N1(C(c2cc(Cl)no2)=O)CCCC1C1CCCN1C(c1cc(F)c(F)c(Cl)c1)=O n1(CC(=O)NC(CN(C)C(c2ccnn2C(F)F)=O)(C)C)cnc(C#N)n1 c1(C(=O)NC2CC(NC(C(CC)OC)=O)C2)cc(C)c2ccccc2n1 C1(CC)CCCN(C(=O)C(C)(C)COCCCC(=O)N(C)COC)C1 C(C(C)C(=O)N1CC(C)(CNC(c2ccc(-c3nn[nH]n3)o2)=O)C1)OC c1(C(N2Cc3c[nH]nc3C2)C(=O)NCC=C)noc2cc(Br)ccc12 N1(C(C2C(COCC)C2)=O)CCC(C)N(C(c2cnc(CC)[nH]c2=N)=O)CC1 C(=O)(C1=C(Cl)CCCC1)N(C(CC)C(=O)NCc1csc(C)c1C)C C1(C(N2C(CCNC(C(c3cnccn3)C)=O)COCC2)=O)CC2(C1)CC2(F)F c1(C(C)(C)OC)nc(C)c(C(=O)NCC(C)N(C)C(C2CC(C)(C)CO2)=O)s1 C(C(=O)NC1CCC(CN(C(=O)CCn2ccnc2C)C)CC1)(C(C)C)OC C1(CCCCC(=O)N(C(CC)CNC(=O)C#CC(C)C)C)SCC2NC(=O)NC12 N1(C(c2cncc(COC)c2)=O)CC2CCC2(CCNC(=O)C(C)(C)CO)C1 N1(C(C(c2ccccc2)C)=O)CCN(CCCNC(=O)CCCCC2CC2)CC1 c1(C(=O)NCCC2OCCN(C(c3cc(C)on3)=O)C2)cnc(C2CC2)nc1C C1(CC)CN(Cc2ccc(-c3cn(CCC(=O)OC)nn3)s2)CCC1CO N1(C(CC(CC)OC)=O)CCc2cccc(O)c2C1 C1(NC(COCCC)=O)C=CCN(C(C2(C)CCN(C)C2)=O)C1 CC(C)(C)C(CNC(=O)COCCCF)NC(c1cc(Br)n[nH]1)=O C(=O)(CC(C)P(C)(C)=O)N1C(Cc2cn(-c3cc(OC)cc(Br)c3)nn2)CCC1 C1(NC(COCC(=C)C)=O)CN(C(=O)C(c2ccc(F)c(F)c2)C)C(C)(C)C1 N1(C(C2CCC(NC(C3CC4CCC3C4)=O)C2)=O)CCC2(CC2)C1 C1(NC(C2CC(CC)C2)=O)CC(=O)N(CCNC(=O)C(C)=C2CCCC2)C1 C#Cc1ccc(C(N2CCC(NC(c3ccc(C)nc3C)=O)C2(C)C)=O)cc1C C1(NC(C(C)NC(N)=O)=O)CC2CCC1(COCCCn1cncn1)C2 c1(C(=O)NC(CCC)CNC(=O)C(O)CN(C)C)ccc2nonc2c1 Cc1cc(C#N)ccc1C(=O)NC1CCOCC1NC(C1CCC(=O)NC1)=O N1(C(COc2ccc(C)cc2F)=O)CCC(C)N(C(c2cc(C#N)c[nH]2)=O)CC1 c1(C(=O)NCCCN(C)C(c2nccc(C#N)c2F)=O)cnc2cccnc2c1 C1(C(N(c2ccn(C)n2)C)=O)CN(C(=O)CC2CCC(O)C2)CCC1(C)C C(C)(CCCC(=O)NCCOC)NC(C(C)OCC=C)=O c1(C(=O)NCCC(C)N(C(c2ccc(C(=O)NC)nc2)=O)C)cc(C)ccc1F C(C(N=c1cc(C)[nH]c(=NCCN2CC=CCC2)[nH]1)c1ccco1)OC C1(C(=O)NCC2C(C(N(C3CC=CC3)C)=O)CC2)CCC(=O)C1 c1(OC)cccc(OC)c1NC(c1cccc(NC(c2c(C)n[nH]c2C)=O)c1)=O c1(C(N(CCCOCCN(C(c2nc(CC)sc2)=O)C)C)=O)cc(N)ccn1 CCCC(CC(=O)N)Sc1ccccc1C#N.c1(C(=O)N)cc(C)ccc1CO N1(C(c2nn(CC)c(=O)cc2)=O)CCC2CCC(C1)N2C(C1CC1C(F)(F)F)=O C1(N(C(C)=O)CCc2nc[nH]n2)(NCc2ccccc2)CCOCC1 N1(C(c2c(CC)c[nH]c2)=O)CCC(NC(c2c[nH]cc(F)c2=O)=O)C(C)C1 N1(C(C(C(CC)C)C)=O)CCOC2(CCN(C(c3csc4cncn34)=O)CC2)C1 CC1C(c2ccccc2)CCCN1Cc1cc(N)ccn1 C1(CCNC(c2cnn(C)n2)=O)(OC)CN(C(c2cnc(C)[nH]2)=O)C1 C1(CC(=O)NC(CC=C)C)N(C(C2CC3CC3C2)=O)CCC1(C)C c1(C(N2CCC(NC(c3c(C)snc3)=O)CC(O)C2)=O)cc(S(N)(=O)=O)n(C)c1 c1(C(=O)NC(C)CCNC(=O)C(C)S(N)(=O)=O)csc2c1CCCC2 C(=O)(N=c1[nH][nH]c2ncc(Br)cc12)C1N(C(C(CC)C(C)(F)F)=O)CC(O)C1 CC1(C(=O)NCC(CNC(=O)CC2CC3(CC3)C2)CO)CCC2(CC1)CC2 c1(C(=O)NCC(C)NC(c2n(CCC)ccc2)=O)cc(C#N)ccc1O C1(CNC(C(C)(C)CNC(=O)CCOC2CCC2)=O)CC(O)C12CCC2 C(CCC(=O)NCc1n[nH]cc1C(=O)NC1C(O)CC1O)NC(N)=O C(N=c1[nH]cnc(NCCCCOC)c1C)n1cc(C(=O)NC)nn1 c1(C(=O)NCCCCC(C)NC(=O)C(C)(C)C2CC2)c[nH]c2ccccc2c1=N C1(C(=O)NCCC(=C)CNC(=O)C(OC)OC)Cc2ccccc2C1(C)C CC1(C)NC(=O)CCC1NC(C1CC(NC(C2CCC(O)C2)=O)CCO1)=O c1(-c2nc(CCS(CC)(=O)=O)nn2CC2CCCC2(F)F)ccc(OC)cc1F N1(C(C(C)CF)=O)CCC(N(C(=O)Cc2cnnn2C)C)CC1 S(=O)(=O)(c1ccc2c(c1)C(=O)N(C)C2=O)Nc1c(COC)cccc1 N1(C(c2c(C)ccc(F)c2)=O)C(CNC(c2csc(S)n2)=O)CC2CCCCC12 C1(C(=O)OC)(C(=O)NC2CN(C(C3CCC(=O)N3C)=O)CC2C)CC2(CCC2)C1 C=CCCCCC(=O)N(C)CC1CN(C(=O)CC(COC)COC)C1 CCCCCC(C)(CC)C(=O)NCC1CCCN(C(C2(C)CSC2)=O)CC1 Cc1cc(C(=O)N(C(C)CN(C(=O)C(F)n2ccnc2)C)C)cc(NC2CC2)n1 C(N=c1[nH]c(=NCCCCN2CCCC2)[nH]c2c1CCCC2)C1NC(=O)C(F)(F)C1 N1(C(c2nc(CCC)oc2)=O)CC(C(=O)N(C2CCC2)C)C(C)(C)C1 c1(C(=O)NC2C3CN(C(CCc4n[nH]c(=N)s4)=O)CC32)nccc2ccncc12 C1(CNC(C(F)=CCC)=O)CCCC1C(=O)NCC(C)(C1CC1)OC C1(CNC(CCCC#C)=O)CC(F)CN(C(=O)CCc2ccc(C)nc2)C1 C1(NC(=O)Cc2ccco2)CCCCN(C(=O)CC(O)c2ccccc2)CC1 C=CC(CC)CC(=O)N1CCSCC1C(=O)NCCc1cn(C)cn1 C1(CNC(C(C)(C)OC)=O)CCCN(C(=O)Cc2cc(F)ccc2F)CC1 C123COC(CN1C(=O)Cn1cc2nn1)C3.C12(C(=O)N)COC(CSC)(C1)C2.CCO c1(OC)ccc(NC(=O)C(O)C2CN(C(C3CC(C)=NO3)=O)C2)c(C)n1 Cc1nc(N2CCN(C(C3CCN(C)C(=O)C3)=O)CC2C)cc2nncn12 C1(CC(=O)NC(CCN(C(c2n(C)nc(C)c2Cl)=O)C)C)CC2(CCCC2)CO1 N1(C(C2CC(NC(C3CC(N(C)C)C3)=O)C2)=O)CCCC1C1CCCO1 N1(C(C(n2cc(COCCCCO)nn2)C)=O)CCC(C)(c2ccc(F)cc2)CC1 c1(CN(C)CC2CCN(C(=O)C(c3ccccc3)F)CC2)ccc(Cl)nc1 C(=O)(C(C)(C)CC(=O)OC)NC1(C)C(NC(C2C3(CC(OCC)C3)C2)=O)CCC1 C(CN=c1[nH]c2ccccc2o1)C1C(C)CCCN1C(C1(C(N)=O)CC1)=O N1(C(CC(=C)C)=O)CC2CCCC(C1)N2C(c1nc2c(CC)cccc2o1)=O N1(C(c2cc(OC)no2)=O)CC(C)CCC1C(=O)N(C)Cc1ccon1 C(=O)(C1=NN(C)C(=O)CC1)NCC(C(=O)NCC(C(=O)OC)C)C N1(C(Cn2c(C)cc(C(F)F)n2)=O)CCC(F)C(NC(C2CCC(=O)C2)=O)C1 C(=O)(C(C(C)(C)C)n1ccnn1)NCC(CNC(C1CC(OC)C1)=O)C c1(NC(CC)CNC(c2cccc(Cl)n2)=O)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] N1(C(C2(OCC)CCC2)=O)CC2CCC1C1CN(C(=O)CN(C3CCC3)C)CC21 C1(CC(=O)NC2N(CC)CC2)CC2(CC2)CN1C(=O)C(CO)OC c1(C(N2CC(N(C)Cc3ccc(O)cc3Br)C2)=O)cc(Cl)nc(Cl)c1 N1(C(C2N(C(C)C)C(=O)CC2)=O)CC2=C(C1)CN(C(=O)CN1CCCC1C)C2 C1(C)(C(N2CCC(NC(C3(COC)CCOCC3)=O)C2)=O)CCC12CCC2 c1(C(N2CC(C)C2C(=O)NOCCC(F)F)=O)c[nH]c(C#N)c1 C(=O)(C(C)(F)C(=O)N1CC2(NC(c3ncccc3F)=O)CCC1C2)OCC Cc1cn2cccc(C(N3CC4CCC4(NC(=O)CCc4nncs4)C3)=O)c2n1 N1(C(CCc2cccc(C)c2)=O)CCOCC12CC(C(=O)O)C(C(=O)O)C2 CCCC(O)(CNC(=O)N(C)OCc1ccccc1)CCC c1(C(=O)NC2CCN(C(C(C)(CO)OC)=O)C2)ccc([N+](=O)[O-])c(C#N)c1 c1(C(=O)NC23CN(C(CN(C)CC)=O)C(C2)C3)cc(Br)cc2c1OCC2 CC(CC(N)=O)C(=O)NCC1(O)CCN(C(=O)CC(C(F)F)n2cccn2)C1 CC(C)CC(O)C(C)C(=O)NCCc1ccsc1C(=O)N(C)CCOC(C)=O S(=O)(=O)(c1ccc(Cl)cc1)N(c1c(F)cnc(C)n1)C1CCCCNC1 c1(C(N2C(CNC(Cc3cccc(C)c3)=O)CCCC2)=O)ccc2c(c1)CC(=O)N2 N1(C(C2ON=C(C(=O)OC)C2)=O)CCC2(CC(NC(=O)CCCCCF)CO2)C1 N1(C(C#CC)=O)CCC2C(CCN2C(c2ccncc2Cl)=O)C1 c1(OCC)cccc(C(=O)OCC)c1O.N12CCC(CC1)NC(=O)C2.C(C)(C)(C)O C=Cn1cc(C(N2CCC(OCC(=O)NC)CC2)C(=O)NCCC#N)cn1 c1(C(=O)OCC)cnc(C(=O)N(C2CCCN(C(C)=O)C2)C)nc1N1CC(C)C1 c1(C(=O)NC(c2cn(CCOC)nc2)=O)ccc(Br)c(C)c1[N+](=O)[O-] c1(C(=O)NCCN(C(C=CC=CC)=O)CCOC)cc(C)c(F)c(C)c1 c1(CC)cc(C)ccc1C(N1CCC(OCCNC(=O)C(C)(C)C(F)F)C1)=O c1(C(=O)NCCC(C(=O)N(C(C)C)CC2CC2)O)ccc2occc2c1 S(=O)(=O)(c1cccc(C(N)=O)c1)NC1(CC)CCN(C(CCCC#C)=O)CC1 C1(N(C)C(c2cc(Cl)c(Br)s2)=O)CCCC2CN(C(=O)C(C)(O)C(F)(F)F)CC12 Cc1cc(C(=O)NC2(C(N)=O)CCCN(C(=O)OC(C)(C)C)C2)nc(C)c1 c1(CC(=O)NC2CC2NC(c2cccc(N3CCCC3)n2)=O)ccc(O)nc1 C1(NC(C)=O)CC(CC(=O)NCCNC(c2cccc(Cl)c2)=O)C1(C)C CS(=O)(=O)CC(=O)N1CCCC1CNC(=O)COc1cccc(O)c1 C(N=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])C1(N(C(Cc2c(C)ocn2)=O)C2CC2)CCC1 N1(C(CC(CCC)O)=O)CC(NC(=O)Cc2ccc3occc3c2)C2(CCC2)C1 c1(CC)cc(C(=O)NC(CNC(c2cc(C)n(C)n2)=O)CC)cc(F)c1 c1(C(=O)NC2CN(C(C3(CSC)CCC3)=O)C2)cnc2c(c1)oc(=O)n2C C(=O)(CS(=O)(=O)N1CCCC1)NCCN(C)C(C1(c2ccccc2)CC1(Cl)Cl)=O C1(CCC(=O)NCCCN(CCC)C(C2CC(=O)N(C)C2)=O)CC(C)(C)CO1 CCCCC(O)CCC(=O)N1CCCC(NC(=O)CN(CC(=O)NCC)C)C1C N1(C(CC)=O)CC(F)(F)CC1(C)CNC(C1CCN(C(C)C)C1)=O CC(C)C(O)C(C)C(=O)N1CCN(C)CC1C(=O)NCC1(C)CC2CC2C1 C1(C(N(CC(C)CNC(C2(CF)CCC2)=O)C)=O)(CC2CC2)CC1(F)F c1(CN2C(=O)CC(COCC)NC2=O)cc2cc(Br)cnc2o1 c1(C(ONC(=O)Cc2cccc(OC)c2Cl)C(=O)OC)cc(F)ccc1OC Cc1ncc(NC(=O)CC2CCCN2C(=O)CCCC2CCCO2)cc1C#N N1(C(=O)Cc2cccc(F)c2)CCCC(C2CCN(Cc3ccnn3C(F)F)C2)C1 c1(OCC(NNC(=O)OC)=O)cc(C)cc(C=O)c1O C1(N(C(C(C2CCC(=O)N2)C)=O)C)CN(C(=O)CCCC(=O)OC)C2CCCC12.CO c1(C(=O)OC)cc(Br)c2nc(NC(c3c(Cl)cnn3C3CCCC3)=O)sc2c1 c1(C(=O)NC(CC=C)CNC(c2c(C(F)F)n[nH]c2C)=O)cc(N)c(F)cc1F C1(C)(NC(Cc2ccc(C)s2)=O)CCN(C(=O)CCc2ccc(C)cc2C)CC1 N1(C(CCOC(C)=O)=O)CCC(NC(c2ncoc2C)=O)CC1C1CC1 N1(C(c2c(C(C)(C)C)ncs2)=O)CC2C(CNC(=O)C(F)n3ccnc3)C2C1 C1(C(=O)NC2CC(C(F)F)C2)(NC(C2CC3CC3C2)=O)CC(CC2CCCC2)C1 c1(CCC)nc(C)c(C(=O)NC2CC(NC(c3conc3C3CCCO3)=O)C2)s1 C1(CC)CCN(C(=O)C=Cc2ccccc2)C(C(=O)NC(C)COC(F)(F)F)C1 C1(COC(C(CCC)NC(=O)OC(C)(C)C)=O)COC2(CCOCC2)CO1 C1(C(N(C)CC2CC(F)(F)C2)=O)CCC(O)CN1C(c1cnc(S)nc1)=O C1(NC(=O)CCN2CCCC2)CCCCCN(C(C2CC2C(F)F)=O)C1 C(CCCCC(=O)NCC1(C(N2CCC(CC)C2C)=O)CCCO1)OCC C(C(=O)NCC(C)NC(=O)CCn1cc(C)cn1)(C(C)(C)C)SC CC(C)C(C#N)C(=O)N1C2CCC1(CNC(c1n[nH]cc1Br)=O)CC2 Cc1csc2ncnc(Nc3cccn4nccc34)c12 c1(CCNC(C2(CCNC(C(C)SCCCC)=O)CCCC2)=O)ncc(C)cn1 CC1=C(c2ccco2)CN(S(=O)(=O)c2cnccc2NCC(CO)C(C)C)CC1 c1(C(N2CCC(C)C(NC(C3CCC(F)C3)=O)C2)=O)cc[nH]c2nccc1-2 N1(CC2C(C)(C)CC2)CCC2(CC1)CC2C(=O)NCCSC1CCCCC1 c1(C(C2(c3cnn(C)c3)C(C)C2)=O)cc(F)c(N)c(F)c1 c1(NC(=O)NC(CC(C)NC(=O)C=CC2CCC2)C)ccc(C(C)(F)F)cc1 C=CC1(C(=O)NOC(c2ccccc2)C)CCN(C(=O)C2=CCSC2)C1 O=C(CCCC(F)F)NCC(CNC(c1cn(CCC2CC2)nn1)=O)CO C1(NC(CC2C(CC)C2)=O)CCCN(C(c2cc(OC)ns2)=O)CC1 C1(NC(c2nc(C(C)C)sc2)=O)CN(C(C2CCCCC2(F)F)=O)CC12CC2 c1(CC(=O)NCC(CC)NC(C(CCC)OC)=O)cccc2c1OCO2 c1(C(c2nnnn2-c2ccccc2)NC(C2CSCCO2)C)ccc(Br)s1 N1(NCc2cccc(C(=O)OC)c2)CCc2c(OC)ccc(C)c2C1 C1(NC(c2cnc(CC)nc2O)=O)CC2CC(C1)N(C(c1ccnnc1Cl)=O)C2 C(=O)(C(C)CCCOC)NC1(CCNC(C(CC)C#N)=O)CCC1 c1(C(=O)NCC(C(C)C)NC(c2cnc[nH]2)=O)ccc2cncc(Br)c2c1 C1(CC(=O)NCc2ccc(CC)s2)CC(C)(C)CN1C(c1nc(C)sc1C)=O C(=O)(C(C)(C)C(F)(F)F)NC(C(C)C)CNC(C1CCC(O)CN1C)=O N1(C(C(C)(C)CO)=O)CCC(O)C(NC(=O)CCc2ccc(F)cc2)C1 C12(NC(C(C)O)=O)CC(CNC(c3c(Cl)cccc3Cl)=O)(C1)OC2C C1(c2nn[nH]n2)(C(=O)NC(=O)C(CSCC)Sc2cn(C)nc2C)CCSCC1 c1(NC(C(CCCNC(C2CCC2(F)F)=O)O)=O)ccc2c(c1)CCC2 c1(C(=O)NCC2C(CNC(COC(C)=O)=O)C2)ccc(C)c2c1CCC2 c1(C(N2CC(N3CCC3)C2)=O)cccc2occc12.C12CCC(C1)NC(=O)CC2 C(=O)(C(O)CCC(F)(F)F)N1CCC(CC=C)(NC(C2CCC(O)C2)=O)C1 C1(NC(C(C)NC(=O)NC2CCCCC2)=O)COC2(CCOCC2)C1 C=CCCCCCCC(=O)N(CCCC(=O)N(CCCCO)CC)C c1(C(N2CC(C)C(CNC(c3cccs3)=O)CC2)=O)ccc2c(c1)nc(O)n2C c1(C(=O)NC(C2(O)CN(C(=O)C(C3CC3)N(C)C)C2)C)ccc(O)cn1 c1(C(N2C(C(=O)NCc3ccc(Br)cc3)CC(O)C2)=O)cc(Cl)cnc1Br C(=O)(CC(C)(C)CC(=O)NC(C)(CNC(C1CC=CCC1)=O)CO)OCC C1(NC(C(C)C(C)S(C)(=O)=O)=O)COC2(CCN(C(c3csc(S)n3)=O)CC2)C1 c1(C(=O)NCC(CC)NC(C(CC)C2CCOCC2)=O)ccccc1COC Cc1cnc(C#N)c(-c2cnc(CC(=O)Nc3ccnc(Br)c3)nc2)c1 c1(NCC(CC)N2CCCC2)nccc(=NCCC(C)c2ccccc2)[nH]1 C12(C(N3CCC(CNC(c4c(C)noc4C)=O)C(C)C3)=O)CCCN(CCC1)C2 c1(C(N2CCN(C(C3(F)C4CCCCC34)=O)CC2)=O)cc2c(F)cc(Cl)cc2[nH]1 c1(C(=O)OC)ccc(F)c(C(N2CC(NC(C34CCCC3C4)=O)CC(C)C2)=O)c1 C(=O)(C(C)C(O)C(C)C)NCC1N(C(CCSCc2cccc(C)c2)=O)CC1 Cc1ccc(CCC(=O)NC2CCC(NC(c3cnnn3C(C)C)=O)C2)cc1C N1(C(c2c(CC)nco2)=O)CCC(CNC(=O)Cn2nc(CC)cc2C)C(C)C1 CC1C(NC(C2OCCO2)=O)CC2CCC1N2C(=O)C(C)OCC1CC1 Cc1nc(-c2ccsc2)ccc1C(N1CCCN(C(=O)NC2CCC2)CC1)=O Cc1cc(C(N2CC(C)(C)CC2CNC(C2CC2(F)F)=O)=O)c(O)cc1F N1(C(C2CC(SC)C2)=O)CCCC1Cn1cc(CNC(=O)CCC2CC2)nn1 N1(C(CC(CCC)(C)C)=O)CCC(NC(=O)C(CC(C)(C)C)OC)CC(O)C1 C12(NC(c3c(C)occ3)=O)CCC(C1)N(C(=O)C(C)NC(=O)C(C)(C)C)C2 C1(c2n(C)ccn2)CN(C(c2sccc2F)=O)CC1NC(=O)Cc1cscn1 c1(NC(C2C(c3n(CC)cnn3)OCC2)=O)cc(C)oc(=O)c1 C1(CNC(CCNC(COC)=O)=O)CN(C(c2cn[nH]c2)=O)C2COCC2O1 c1(OCC)nccc(C(=O)NC(CNC(c2ccc(Br)cc2C)=O)CO)c1F C(CC(F)F)(C(=O)NCC1C2CCCC12)N(C(c1c(CC)cncc1)=O)C C12(C(=O)NC3CCC(CNC(C(=O)N(C)C)=O)C3)CC3CC(C1)CC(CO)(C3)C2 CCC(CN(C(=O)CC(=O)OC)C(c1nc(C)oc1C)C)C(=O)OC(C)(C)C CC(C)CC(C(=O)N(CC(O)CN(C)C)C)ONC(=O)CCn1cccc1 c1(C(N2CCCC2c2cn[nH]c2)=O)csc(-c2ccc(CO)o2)n1 c1(CCC)nc(C)c(C(=O)NCC2CCCN(C(=O)CC(C)n3ccnc3)C2)s1 c1(-c2cn(-c3ccc(C(N(C4CCOC4)CC)=O)cc3)nn2)c(Cl)cccc1Br Cc1nnccc1C(=O)NCCN(C(C1CC2CCC1O2)=O)CC1CC1 N1(C(c2cc(OCC)ncc2)=O)CCCC2(NC(C3CCC(C)(C)O3)=O)CC2C1 C1(NC(C(=O)NCCNC(C)=O)=O)CCC(N(C)C)C1 C12(C(=O)NCC3(C)N(C(C(C)C#N)=O)CCC3)CCCCC(=O)N1CCC2 C(=O)(C#CC1CC(F)(F)C1)NCC(CCNC(c1c[nH]nc1C)=O)OC N1(C(c2ccc(N(C(C)C)C)cc2)=O)CCC(CO)(NC(=O)C=C2CCC2)CC1 C(=O)(C1=CC2(CCOCC2)C1)N1CC(C(C)NC(CCc2ccc(C)s2)=O)C1 N1(C(C(CO)OC)=O)CC(C(=O)NC2COC(C)(C)C2)C(C)(C)C1 CC1(C)C(CC(N2CCCC(CC(=O)NCC3CC4(CCC4)C3)C2)=O)C1(C)C CC1CN(C(=O)C(CNC(C2(C#N)CC(=O)C2)=O)CC2CC2)CCO1 c1(CC)noc2ncc(C(=O)NC34CCCN(C(c5cc[nH]c5)=O)CC3C4)cc12 C(=O)(C(C)N=[N+]=[N-])N(C(C)C(=O)NC1C(C)C1C)CCC c1(C(=O)NCC2CCCCC2NC(C23CCC(CC2)O3)=O)nccc2[nH]ccc12 C(=O)(CC(CNC(c1ccccc1Cl)=O)OC)N(CC)Cc1noc(C)n1 C(CCCC(=O)N1CCCC(CN(C(=O)COCc2ccnn2C)C)C1)SC c1(CN2CCC(C(C(=O)NCC)NC(=O)OC(C)(C)C)CC2)ccc(F)cc1F C(c1ccc(N)o1)=CC(N1CCC(CNC(C2(COCC)CC2)=O)C1)=O.CC c1(N(CCSC)C)[nH]c(=NCc2cc(Cl)nc(=N)[nH]2)nc2scnc12 C1(O)(CC(=O)NCCC2CCCN(C(C(CC)(C)O)=O)C2)CCCCCC1 C1(NC(C2CC3(CC(=C)C3)C2)=O)C(C)CCN(C(c2cc3n(n2)CCCC3)=O)C1C N1(C(=O)OC)CCCC(NC(=O)C(n2cc(CN(C)C3CC3)nn2)C)C1 C(C)(N=c1[nH]ccnc1F)C1N(C(c2c(CC)ccc(C)c2)=O)CCCC1 C1(CCNC(c2ncoc2Cl)=O)CCCCN1C(C1C=CCCC1)=O C1(CN(C(C2C(C=C)C2)=O)CC)CC12CCN(C(=O)C(O)Cn1cncn1)CC2 C1(C(N2CC(CNC(c3sc4ncn(C)c4c3)=O)C2)=O)CCCCC12CC2(F)F C1(NC(C=C(C)Cl)=O)CC2CC(NC(=O)CC3CC4CC4C3)C2C1 C1(C(=O)NC2CCCC2C(=O)Nc2cncc(Cl)n2)CCc2nc[nH]c2C1 C(=O)(C(CC)CCCC)N1CC2(CN(C(CC3(C=C)CCC3)=O)C2)C1 c1(NC(C(=O)NCC2CC2)=O)ccc(CCNC(C(CC)NC(N)=O)=O)cc1 n1(CC)ccnc1C(C)NC(=O)C(=O)Nc1nc(C2CCCCC2)ns1 c1(C(N2CCCCC(CO)C2)=O)cc(C(C)C)cc(C(F)F)c1 c1(C(N(C2CN(C(=O)C3=NNC(=O)CC3)C2)C)=O)cccc2c1OCCC2 c1(C(N(CC(=O)NC2CCCC2)C(C)C)=O)cnn[nH]1.C(CO)N Cn1nnc2cc(C(=O)NC3(C4CCCN4C(C4CCCN4C)=O)CC3)sc12 C(C1COC(C)(C)O1)=CC(=O)NC(C)CNC(C1CCCOCC1)=O O=S(=O)(c1cn[nH]c1)N1CCC(NCc2cccc(Cl)n2)C(F)C1 C1(C)(CNC(c2cnc(C(C)(C)C)[nH]2)=O)CCN(C(C2(Br)CC2)=O)CC1 c1(C(N2CC(COC)(NC(C3COC(C)C3)=O)C2)=O)ccc(F)c(C(F)F)c1F C1(CNC(Cc2n(C)nnc2)=O)CCC(C(=O)NCCCCCCF)CC1 CCC(CNC(=O)C(C)Nc1ccccn1)(CC)NC(=O)Cn1nc(C)cc1C c1(C(=O)OC)cnc(N(C)C(=O)NC2CCC(C)C2)c([N+](=O)[O-])c1 CCC(CCCC(=O)N1CCC(F)(C(N)=O)C1)NC(c1nc(C)oc1C)=O c1(CC(=O)NC2C(NC(C(CC=CC)CC)=O)CC2)c(C)[nH]c2ccnn2c1=O C(=O)(C1CCCc2c1ncn2C)NC(C1N(c2nnc(C)s2)CCC1)(C)C N1(C(c2n(CC)nnc2)=O)CC(CNC(c2ccc(C)c(C)c2)=O)OC(C)(C)C1 C(=O)(CCCCC1CCC1)N(C(=O)COC1(C)CCOCC1)CCOC c1(OCC(=O)NC(C(CO)NC(CC=C(C)C)=O)C)c(C)cc(Cl)cc1C c1(C(N(CC(O)CN(C)C(C2CCCC2CF)=O)C)=O)cc(C(N)=O)cc(F)c1 Cc1nc(N2CCC(C)(C)C(CNC(c3ccc(O)nc3)=O)C2)c2cc[nH]c2n1 c1(C(=O)NCCN(C(CC(C)OC)=O)CC2CC2)c[nH]c2cc(C)ccc12 N1(C(CCC)=O)CC(C)CCC1CNC(=O)CCc1ccc(OC)c(C)c1 c1(C(N(C(c2ccccc2)CNC(CC2CC(C)C2)=O)C)=O)ccc(=O)n(C)c1 C(C(C(=O)NC(C(C)C)C(C)C)C(C)(C)C)NC(c1cc(CC)sn1)=O N1(C(CC2N(C)CCC2)=O)CCC(F)C(C(F)(F)F)C1.CCSCO c1(NC(C)=O)ccc(C(=O)NCC(O)CNC(C2CCCCN2C(N)=O)=O)cc1 C1(NC(c2c(C)n(C)cn2)=O)CC2CC(NC(C3CC3c3ccccc3)=O)C1C2 CC(C)(C#N)CCCC(=O)NCCNC(C1CCOC1)=O c1(N2CCCC(C(=O)Nc3ccc(F)nc3F)C2)nc(CO)nc2ccccc12 c1(C(=O)NCCCNC(=O)Nc2ncccn2)cnc2c(c1)CCC2 C=C1CC2(C1)CN(C(=O)C(F)CC1CN(C(C3CC3=C)=O)C1)C2 C1(CNC(C(C(C)C)O)=O)Cc2ccccc2CN1C(C1CCC(=O)N1)=O C1(NC(C(CO)N(C)C)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1CO C1(NC(C(CCC)OC)=O)CC2CCC(C1)N2C(C1CCCCC1OC)=O N1(C(CONC(c2c(OC)nccc2)=O)=O)CC(CO)C2(CC2)C1 C1(C(=O)NC(C(=O)OCC)C(C)(C)C)CC12CCN(Cc1c[nH]c(Br)c1)CC2 C1(CC)CCCCCCN1C(C1CCN(C(c2csnc2Cl)=O)C(C)C1)=O N1(C(c2cn(C)nc2O)=O)CCC(CO)(CNC(C2(O)CC2)=O)CC1 N1(C(c2ncc(C)c(Cl)c2)=O)CC(NC(C2CNC(=O)C2)=O)Cc2ccccc21 C1(CC)CCC(C(=O)NCCCN(C(c2cc(Br)n[nH]2)=O)CC)O1 Cc1cc(F)c(CNC2CCN(C)CC2C)cc1[N+](=O)[O-] c1(C(C(=O)N(C(C)CNC(c2ccc(F)s2)=O)CC)C2CC2)ccc(C)cc1 C1(C(=O)NCC2(CC)CC2)(COC)CCCN1C(=O)C=CCCC(C)C C1(NC(C(C)CO)=O)CN(C(c2cc(C3CC3)cs2)=O)C2(CCC2)C1 c1(C(=O)NCC2N(C(C3C(CC)C3)=O)CCC2)cnccc1Cl CC1C(O)CCCN1C(=O)CCCN(C)C(c1coc(C2CC2)n1)=O c1(C(=O)NCC2CC(NC(C3CC(O)C(F)C3)=O)C2)cc([N+](=O)[O-])cnc1O N1(C(C2(OCC)CCC2)=O)C2CCCC1CN(C(C1CC(C)=NO1)=O)C2 c1(C(N2CCCC(NC(C3(C)ON=C(C)C3)=O)CC2)=O)cnc2nccnc2c1 C1(NC(C(C2CCOC2)OC)=O)CCCCC1n1cc(Cn2cc(CO)nn2)nn1 C(CCCCC(=O)N1CCCN(CC)CC1)N(C(C1(CCCC)CC1)=O)C CN=c1cc(C(N2CC(C(N3CCOC(C4CC4)C3)=O)C2)=O)cc[nH]1 CC1(C)CCCC(C(N2CCCC3(NC(=O)CCc4cscn4)CC3C2)=O)CC1 N1(C(C2=C(C)CC2)=O)CC(NC(=O)C(C(C)C)NC(=O)C(F)(F)F)C(C)(C)C1 C=CC(O)C(=O)NC(CN(C)C(c1cnc(N(C)C)o1)=O)Cc1ccccc1 c1(C(=O)NC2CC(C(=O)Nc3c(C(N)=O)ccc(F)c3)C2)cc(F)c(Br)cc1Cl c1(C(=O)NC(CNC(CN(c2cnccn2)C)=O)C2CC2)cc2n(n1)CCCC2 CCCC(CCC)CC(=O)NC1C(C)CN(C(c2ccsc2)=O)CC1C c1(C(N2CC(C)(NC(c3cc(CCO)on3)=O)C2)=O)[nH][nH]c(=N)c1Br N1(C(C2(C)CCC2)=O)CCCC(O)(CNC(c2cncc(C#N)c2)=O)C1 CC1OC2(C(=O)NCC3(CNC(c4ccncc4O)=O)CCC3)CC1C2 CC(C)CC(CNC(c1cn(C)c(=O)n1C)=O)C(=O)NCC1CC(C)(C)C1 C=CC1COCCN1C(C1CN(C)CCN1C(c1cc(C)c(C)o1)=O)=O n1(CC(=O)NC2C(C)CCN(C(c3ccccn3)=O)C2)nc2ccccn2c1=O Cn1ncc(C(=O)NCC2CN(C(=O)CC3CC3)C3(CCC3)C2)c1S(N)(=O)=O N1(c2ccn(C)n2)CCCC(NC(c2cn(C3CCCCC3)nn2)=O)C1=O CC(C)C(C(=O)NCC(CNC(=O)C(CO)N(C)C)CO)C1CC1 C(C)(C(=O)N(C)CCOCCNC(=O)CSC1CC1)(C1(C)CC1)OC c1(C(=O)OCC(N2CC(C#C)OCC2)=O)ccc([N+](=O)[O-])nc1 N1(C(CC=C(C)C)=O)CCCC(C)(CNC(c2cc(-c3ccco3)on2)=O)C1 C1(NC(C(OC)OC)=O)CCN(C(C2(C(C)C)CC2)=O)CC1C c1(C(=O)NCC2(CCNC(C(CC)O)=O)CC2)cc2c(s1)CCC(CC)C2 Cc1ccc(CNC(=O)CCNC(=O)CN2CCC(=O)CC2)c(F)c1 C1(NC(c2ncc(CC)nc2)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CC2(CC2)C1 N1(C(C(C)CO)=O)CCCN(C(c2cc(C3CCCO3)n(C)n2)=O)CCC1 c1(N(CCCNC(c2ccc(CN3CCOCC3)o2)=O)CC)ncnc(=N)[nH]1 CC1CN(C(=O)CCCCNC(N)=O)CCC1CNC(c1cnn(C)c1Cl)=O CCCCC(C(=O)NCCC[Si](C)(C)C)NC(c1ccccc1CC#N)=O Cc1cccc(C)c1N1CCC(NC(=O)C(CCO[Si](C)(C)C(C)(C)C)C(C)C)CC1 CCCCC(C)C(=O)N(CCNC(=O)CCCC(=O)NCC1CC1)C(C)C Cc1nc2c([nH]1)CC(C(=O)NCC1(O)CCN(C(c3n[nH]c(C)c3Cl)=O)C1)CC2 C1(CC(N2CCC(F)(CNC(C(CCC)=CCC)=O)C2)=O)NC(=O)CN(C)C1=O N1(C(c2cc(C)[nH]n2)=O)CC(CNC(=O)CNS(N)(=O)=O)CC12CCC2 c1(NC(C(=O)NCC2(C)CCCS2)=O)cc(F)ccc1Cl c1(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)OC)ncc(C)cc1C C(=O)(CCCCC(=O)O)NC(Cn1cc(-c2cccc(C)c2C)nn1)CN(C)C Cc1ccc(NC(=O)C(C)Sc2ccco2)cc1S(=O)(=O)Nc1ccc(Br)cc1 c1(CC(N2CCC(C)(NC(C=C(CC)CC)=O)CC2)=O)nc2cccc(F)c2[nH]1 c1(C(N2CCC(OCCF)C2)=O)cn(CCNC(=O)C(F)n2ccnc2)nn1 C1(F)(CNC(C2(C)CCC2)=O)CC(NC(=O)C(=O)NCC(F)(F)F)C1 c1(C(C)(C)C)ccc2c(c1)C(NC(c1ccc(F)c(Cl)c1)CBr)CC2 C1(C(=O)NCC2CC(F)(F)C2)CC2(CC2)CN1C(c1cnsc1)=O Cc1nc2c(N3CC4CCC(C3)N(S(=O)(=O)CC3CC3)C4)ncnc2[nH]1 N1(c2ncnc(NC(c3ccco3)CC)c2C)CCCC2(CCOCC2)C1 C1(NC(C(CCNC(=O)CCc2nccs2)OC)=O)CCCC12CC2 c1(C(=O)NC2CN(C(Cc3scc(C)c3)=O)C(C)C2)sc2nnc(S)n2c1C N#Cc1ccc(C(=O)NC2(CNC(C3Cc4cscc4C3)=O)CCCC2)c(F)c1 CC1CCN(C(=O)CCCc2ccsc2)CC1NC(=O)Cc1ccon1 C(=O)(C(C)(C)CO)NCCOCCNC(c1[nH]cc(C(=O)OC(C)(C)C)c1)=O C1(C)(C(=O)NC2C(C(=O)NC(c3nc(=O)o[nH]3)C)OCC2)CCCN1C c1(N2CC(=C(CN(C(=O)C=Cc3ccc(Cl)cc3)C)F)C2)cc2nncn2cn1 N1(C(C(C)SCC)=O)CCOCC(CNC(c2ccc(=O)n(O)c2)=O)C1 c1(OC)ccc(C(=O)NCC(O)CNC(c2cccc(O)c2Cl)=O)c(Cl)n1 C(C(=O)NC1(C(N2CC(N3CCOC3=O)C2)=O)CCN(C)C1)(C(C)C)SCC N1(C(c2cc(CC)ncc2)=O)CC2CCCC(NC(c3ccc(O)nn3)=O)C2C1 S(=O)(=O)(c1cnc(Cl)n1C)NCCCC(=O)N(C)C C(=O)(CC(C)NC(=O)CCc1cnn(C)n1)NCC(CNC(N)=O)OC C1(NC(c2cnc(CC)s2)=O)C2CC3C(C2)C13C(=O)NCc1ncc(O)cn1 CCC(C(=O)NC1CCC(N(C)C(c2nccnc2N)=O)CC1)C(C)(C)CC N1(C(C2(COC(C)CC)CC2)=O)CC(NC(COCCCOC)=O)C1 C1(CNC(C(C2CCC2)NC(C)=O)=O)CN(C)CCN1C(=O)CCC1(C)CC1 c1(COC)cncc(C(=O)NC2(CNC(C3(C)CC3(F)Cl)=O)CC2)c1 C1(SC)CN(C(=O)Cn2cc(CN3CC4CC4C3)nn2)CC12CC2 N1(C(c2cnsc2NC(=O)C(c2ccc(O)cc2)OC)=O)CCCC(O)C1.CC C1(C(N2CCC2Cc2ccccc2)=O)(CNC(C2CC(OC)C2)=O)CCCO1 N1(Cc2cccc(F)c2)CCc2ccccc2C1.c1(CC(=O)N)csc(CO)n1 CCC(C)(C)C(C)CC(=O)NC1CN(C(c2ccc(Br)c(F)c2C)=O)C1 C=CCC(CC=C)C(=O)NC(C(=O)NC(C)Cc1nncn1C)C1(C)CC1 c1(C(=O)NCC(N(C(=O)CC2CC2(Cl)Cl)C)C2CC2)ccn(CC(F)(F)F)n1 CON1CCC(C(=O)NC2CCCC2CN(C)C(C2(C)CC3CCC2O3)=O)CC1 c1(C(N(CCCNC(c2scc(C)c2Cl)=O)CC)=O)cc2c(C)cc(F)cc2[nH]1 C(c1ccccc1F)=CC(=O)N(CCCCCC)CCNC(=O)CC1(O)CCC1 C(=O)(C(C)(C)CN1CCCCC1)OC(C)(C)C.N1(C(C2(CO)CC2)=O)CCCC1C N1(C(c2c(C)ncc(S(N)(=O)=O)c2)=O)CCC(C2CCCN(CC#N)CC2)CC1 C#CCCN=C(NCc1nc(C(C)(F)F)cs1)N1CC(C)CC(C)(C)C1 C(C(O)CCNC(C1CCCC1C)=O)NC(C(OCC)OCC)=O Cc1nc(-n2nc(CCCO)nc2-c2cscc2Cl)n(C)n1 C(=O)(C(C)CCNC(C1CCC(C)N1C(=O)Cn1cnnc1O)=O)OC C1(NC(C(C)Cc2cnc[nH]2)=O)CCCCN(C(=O)Cn2cccc2)C1 CC1CCCN(C(c2cnc(CNC(=O)CCS(C)=O)nc2)=O)CC1 N1(c2c(OC)cnc(Cl)n2)CCCC2(NC(c3cnc(C)[nH]3)=O)CC2C1 Cc1ccc(C(N2CC(CN(C)C(C34CCC(C)(C3)OC4)=O)C2)=O)nc1F Cc1cc(NC(C2CC(C)(NC(=O)CSC(F)(F)F)C2)=O)c(Cl)cc1Cl S(=O)(=O)(c1cnn2ccc(=NCC(c3cccs3)N(C)C)[nH]c12)NCC#CC C(C)(C)(C(=O)NCC(C)CNC(=O)CN1CC2CC2C1)OC(C)C C(=O)(CCCN(C(=O)CCCNC(C)=O)C)NC(C(=O)OC)C N1(C(C=CCC)=O)CC(C)(C)OCC1CNC(=O)C(C)c1cc[nH]n1 C1(C(=O)NC2CC(CCNC(c3ccsc3Cl)=O)C2)CC2CC2C1 O=C1CC(C(=O)NC(Cc2cc[nH]n2)C(=O)NCC2CC23CCC3)CC(=O)N1 N(C(=NCCC(C)(C)OC)NCc1cnc(C)s1)CC(=C)C c1(C(c2nnnn2CCCF)NC(C(=O)N(CC)CC)C)sc(Br)cc1C C1(NC(=O)C=C(Cl)Cl)COC2(CCN(C(c3ncc(C4CC4)cc3F)=O)C2)C1 C(CC(C(=O)Nc1cnc(SC)nc1)NC(=O)C(F)F)OCC c1(C(N2C(C)(CNC(c3ccc(Br)o3)=O)CCC2)=O)nc2ccccn2c1F C(=O)(CCCOC(C)(C)C)NCC=CC(C)NC(CSCCCC)=O c1(CC(=O)NCC(C2CC2)NC(C2(C)CCCCO2)=O)cccc2[nH]ncc12 Cc1ccc(C=CC(=O)N(C(C)CNC(c2ccc(C(F)(F)F)s2)=O)C)cc1Cl C1(CNC(C2C(C)(C(F)F)C2)=O)(NC(c2cnc(Cl)[nH]2)=O)CCCC1 N1(CC(N2CC(n3cc(CC(OC)OC)nn3)C2)=O)OC(C)(C)CC1=O C1(NC(C(CN(C)C)NC(CCNC(C)=O)=O)=O)CN(C)CCC1O c1(C(N2CCC(NC(COC)=O)C23CCC3)=O)cc2c(o1)C(C)(C)CCNC2=O C(=O)(C1=C(Cl)CCOC1)NCC1N(C(C(C)CC(F)F)=O)C2CCC1C2 c1ccc2c(c1)CCCC2CN(c1ncccn1)Cc1ccc2c(c1)OCCO2 C(=O)(C1=CCSC1)NCCC(=C)CNC(c1csc(C(N)=O)n1)=O c1(C(N(CCOCCN(C(=O)Cc2ccsc2)C)C)=O)cccc2c1COCC2 c1(C(=O)NC(CC)CN(C(=O)CC(C)C(C)C)C)ccc2cnsc2c1 Cc1ccc(C(N2CCCCC(CNC(=O)Cc3nccn3C)C2)=O)c(C)n1 C1(C(N(CCC(F)(F)F)CC)=O)CCCCN(C(c2cccnc2)=O)C1 c1(NC(C(C)C)CCN(C(=O)CC(C)CN(C)C)C)c(Cl)cncc1[N+](=O)[O-] C1(CNC(c2ccc(OCC)cc2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1C c1(C(N(CCNC(c2ccc3c(c2)CC3)=O)C2CC2)=O)ccc2occc2c1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCC(C2CN(C(=O)CCS(C)=O)C2)C1 C1(CNC(CC(C(C)C)C)=O)CN(C(=O)Cc2ccns2)CCC1(C)C N1(C(c2ccc(SCC)cc2)=O)CC(NC(=O)C(CC)OCCOC)CC(O)C1 c1(NC(N2C(c3cc(C(=O)OCC)no3)CCCC2)=O)nccc(C(F)(F)F)c1F C(=O)(C(C)(C)C(=O)Nc1ncnn1CCF)NC1CCCC(COCC)C1 CCC(CCC(=O)Nc1cnn(C)c1C)NC(c1cocc1C)=O Cc1nnc2n1CC(C(N1CCC(N(C)C(c3cc4ccccn4n3)=O)C1)=O)C2 S(=O)(=O)(c1cc(Br)ccc1OC(C)CS(C)=O)NC1CC(NC(=O)OC)C1 C(=O)(N=c1ccc([N+](=O)[O-])c(Br)[nH]1)NC(C1CCCCO1)C Cc1nc(N2CCC(NC(=O)C=CCF)C(CO)CC2)ccc1[N+](=O)[O-] N1(C(C(CCC)N(C)C)=O)CCOCC(NC(=O)CCc2ccn(C)c2)C1 C1(C(=O)OC)C2C=CC(CC2)C1C(=O)NCC1(c2nn[nH]n2)CCOC1 CC(C)(C)C(O)CCC(=O)NC1CC(CNC(C23CCC(C)(C2)OC3)=O)C1 c1(C(C(=O)NC(C)CCNC(=O)CSC(F)(F)F)(C)C)cccc(Cl)c1 c1(C(=O)NC2C(NC(c3ccc(Cl)s3)=O)C2)cnc2n1CCCC2 C1(CNC(C2C(C(=O)NC3CCC(C(=O)OCC)CC3)C2)=O)CCC(C)(C)OC1 C1(CC(=O)NC2CCN(C(=O)C=Cc3cccnc3)CC2)CCCC(=O)N1 N1(C(C(CCC2CC2)NC(C2C(CC)CCCC2)=O)=O)CCC(C)(C)CC1 N1(CC(C)Cc2ccc(OC(F)F)c(Cl)c2)C(=O)N(CCF)C(=O)C12CCCC2 c1(NCC2C(NC(=O)OC(C)(C)C)CC2)ccc(CO)o1 N1(C(C2C(=C)C2)=O)CC2CC(C(=O)N(C3CN(C4CC4)C3)CC)C(C2)C1 CC(CNC(=O)CCc1cncs1)(CO)NC(=O)CC1(C)CCOC1 NC1(C(=O)Nc2nccn2Cc2ccccc2)CC(C2CCC2)C1 CCC(C)CCCCC(=O)NC1CC2CN(C(=O)C(F)(F)CC3CC3)CC2C1 C(=O)(C1c2ccoc2CCN1C(CC)C(=O)NC)OCC C(=O)(C(C(C)(C)C)NC(=O)Cc1cn[nH]c1)N1C(CSC)CC(OC)C1 C(CC(=C1N=NNN1c1ccccc1)NC(c1ccccc1)CN)S(C)(=O)=O Cc1ccc(C(N2CCC23CCC3)=O)c(N)n1 C1(C(=O)NCC2(NC(COCCCC)=O)CC2)Cc2nccn2C1 C1(CC)CN(C(=O)CNC(c2ccccc2)=O)CCN1C(c1cn(CC)cn1)=O C(=O)(CCS(N)(=O)=O)N1CCCC(N(C(Cc2c(C)n(C)cn2)=O)CCO)C1 c1(OCCC)ccc(S(=O)(=O)N2CCC(NC(c3ncsc3C)=O)C2)cc1 CC1OC2CCC1(C(=O)NCC1(NC(C3CN(S(=O)(=O)C(F)F)C3)=O)CC1)C2 C(=O)(C(O)CCNC(=O)C=C(C)c1ccco1)NC(C#C)(C)C1CCCC1 C(=O)(C(F)C(C)CNC(C1CC2(CCC2)CO1)=O)NCc1ccc(C)s1 CCCCC(CNC(=O)CCOc1cccnc1)NC(=O)CCOCC(F)F C(C(F)(F)CC(O)CO)N(C(c1ccc(-c2ccc(C)cc2)o1)C(=O)NC(C)C)C c1(C(N(CC(C)NC(C(CC=CC)CC)=O)CC)=O)cc2c(ncn2C)n1C N1(C(C(CCC2CCC2)NC(c2c(C)csn2)=O)=O)CC2(C=CCO2)C1 c1(CN2C(CNC(C(C)c3cccs3)=O)COCC2)cc2ccccc2nc1O C(=O)(CCC(=O)NC1CC2(C1)CC2NC(=O)CCn1cnccc1=O)NCC c1(C(N2CC3(CC(NC(=O)CO)C3)C2)=O)cn2ccnc2cn1 C1(C(=O)NC(C)CNC(C2CC(n3cnnc3)C2)=O)CCOCC1(C)C c1(C(=O)NC2CCN(C(CC(CC)O)=O)CC2F)cc(Br)cc2c1cnn2C n1(CC(=O)NC2CCCC(NC(c3cc(OC)ncc3)=O)C2)nc(O)ccc1=O CC(C)S(=O)(=O)CC(=O)N1CC(CNC(=O)CC2CCCCN2C)C1 N1(C(CCN(C)CC)=O)CCOC(C(N2CC(COC)C2)=O)CC1 c1(CC(CN(C)Cc2cc(C3CC3)n[nH]2)=O)ccc(C(F)(F)F)cc1 O=C(C1=CCCS1)NCc1ccc(CCNC(=O)CC2CCNC(=O)C2)cc1 c1(CNC(CSc2n[nH]c(=N)s2)=O)ccnc2c1CCO2.C12CC(C1)NC2=O C1(CNC(C2(C(N)=O)CCC2)=O)CCCC(CNC(C2CC23CCC3)=O)C1 C(=O)(CCP(C)(C)=O)NCCCCNC(C12CC(C(=O)OC)(C1)C2)=O c1(C(=O)NCC2CC(OC)C2)[nH]ccc1CNC(C1(N(C)C)CC1)=O CC(C)C(COC)C(=O)NC1(NC(=O)C(C)ONC(=O)OC(C)(C)C)CCOCC1 N(C(=NCCC1(CO)CC1)NC1CC1(C)C(F)(F)F)C(C1CCCO1)C C(=O)(N1CCC(C(N2CCC2CC2CC2)=O)O1)C1C(C)CC1 c1(C(=O)NC2CCCN(C(C3(N(C)C)CCC3)=O)CC2)cccc2c1OCO2 C1(C(N)=O)CCC(C(=O)NCCC2CC(NC(=O)CCCn3cccn3)C2)CC1 c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)c(O)cnc2ccccc12 C(=O)(CCC1=CCCCC1)NC(C(C)C)CC(=O)NCCc1ccccn1 c1(C(=O)NC2CCCN(C(C)C)C2)cnn2c1CN(C(=O)OC(C)(C)C)CC2 C1(CC(=O)NC2(CN(C(c3cc(C)no3)=O)C)CC2)CC(C)(C)OC1=O C(=O)(CCCCCC(C)O)N(CCCNC(C=COCC)=O)C(C)C N1(CCCCN2C(=O)NC(C)C2=O)CCN(C)Cn2nnnc21 S(=O)(=O)(c1cnn2ccc(NC3CC4(CC4)C3)nc12)N1CC(C)SC(C)C1 c1(C(N2CC3=C(CN(C(C4CCN(C)C4)=O)C3)C2)=O)cnn2c1OCC(F)C2 c1(N2C(=O)CC(NC(c3n(C)c(C(F)F)nn3)=O)C2)ccc(Cl)c(Cl)c1 C(=O)(CCCCCSC)N(C(CCNC(C1C(COC)(CC)C1)=O)C)C C(=O)(CCCC(=O)NC1CC2(C1)CC(NC(C1CCOC(C3CC3)C1)=O)C2)OC c1(OCC(N2CCCC(CC(=O)Nc3ccccc3)C2)=O)c[nH]nc1[N+](=O)[O-] N1(C(C2CC2C(=O)Nc2c(OC)c[nH]n2)=O)CCCC(F)(F)CC1 n1(CC(=O)NCC2(C)CCN(C(=O)C3=CCC3)CC2)c(=O)oc2ccccc12 C(CCC(C)(C)C(=O)Nc1cccc(O)c1)NC(CC1C(C)OCC1)=O c12ccc(cc1)CNC2.c1(NC(c2nc(C(C)C)oc2)=O)cncnc1Cl N1(C(C(C(CC)C)=O)=O)Cc2ccc(C(C)NC(=O)CCCC)cc2C1 N1(C(c2c(OCCCC)cccc2)=O)CC23COCC2(C1)C3 CCCCC(CC)CC(=O)NCC1CN(C(=O)COC2(C)CCC2)CCC1C CC(C)CCCCC(=O)NC1CCC(CNC(=O)Cc2cnns2)C1 C(=O)(C(CC(C)C)ONC(=O)C=C=C(C)C)NC(COC)CCO c1(C(C(N2C(CNC(CC(=O)NCC)=O)CC(OC)C2)=O)=O)cc(F)ccc1C Cc1cnc(C)c(C(=O)NCC2C3CC3CN2C(=O)C(C)N(C)C)c1 C(=O)(C(C)(C)C(=O)NCC1CC2(CC(NC(=O)C(C(C)C)N(C)C)C2)C1)OC N1(C(=O)OC)CCCC2C1CCN2C(=O)Cn1cc(C(F)(F)F)ccc1=O.C(=O)(O)O N1(C(COC2CC(CNC(c3c(C)nns3)=O)C2)=O)CCC2(COC(=O)N2)C1 c12ccccc1Cn1cc-2nn1.CC1(C(=O)NCC2(O)COC2)CC1Br c1(SC)ccc(NC(C2CCN(C(=O)C(N)=O)C2C)=O)cn1 c1(C(c2n(CC)nnn2)NC(Cc2ccccc2)C(N)=O)cnc2n1CCOC2 c1(OCC)cc(CNc2cccnc2NC(c2cnccn2)=O)cc(Br)c1O c1(SC)cc(C(N2CCOCC2CN(C(=O)C(C)n2cccn2)C)=O)c(C)o1 C1(CNC(CSCCC(C)C)=O)CN(C(=O)CCC(C)(C)N(C)C)CC1(C)C N1(C(c2n(C=C)ncc2)=O)CC(NC(c2cc(Cl)n[nH]c2=N)=O)CC(F)(F)C1 N1(CC(=O)NCCN(C(c2ncc(C)s2)=O)CC)CCCC1=O [N-]=[N+]=Nc1ccc(C(N2CC3C(CNC(C4CCSC4)=O)C3C2)=O)cc1 c1(N(C)C)ccc(F)c(C(=O)NCC(O)CNC(=O)CSc2cccc(Cl)c2)c1 N1(C(COCC=C)=O)CCCC(NC(C2C(C)C2(F)F)=O)CC1 c1(NC(c2n(CC)nnn2)C(C)C2CC2)ccc(C(c2ccccn2)OC)cc1 c1(OC)ccc(C(N2CCC3(NC(=O)CCCC(C)=O)CC3C2)=O)cc1OC Cc1nn(C(C)(C)C)cc1C(=O)NCCOCCCN(C)C(C1CC=CC1)=O C(=O)(CC1OCc2ncccc21)N(C(C#C)COC)C C1(NC(C2CCCOC2)=O)C=CCN(C(=O)Cc2nnc(S)n2CCO)C1 c1(NC(c2nc3ccccc3o2)C)[nH]c(=NCCc2nccs2)nc2sccc12 CC(C)(C(=O)N1CC2CCC1C(NC(=O)C=Cc1ccc(Cl)cc1)C2)C(F)(F)F O=C(C1=CC2(CN(C(c3nc(Cl)cs3)=O)C2)OC1)NCC(C1CC1)C1CC1 C1(CNC(CCc2cnn(C)n2)=O)CCCCC1NC(c1cc(C(F)F)[nH]n1)=O C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1CCC(NC(C2N(CC)CCOC2)=O)CC1 n1(CC(=O)NC2CCN(C(C(C)(C)n3cccn3)=O)C2)cnc(C#N)n1 C1(C(=O)NC(CCSC)CO)CC2(CC2)CN1Cc1cc(Br)ccc1O C1(CC(=O)NCc2c(C(C)NC(C)=O)cccc2)Oc2ccccc2NC1=O c1(C(N2CCC3(C(C(N4CC(OCC)C4)=O)C3)C2)=O)ccc(F)cc1C CC1(C)CCN(C(=NCCC(=O)N2CCCCC2)NCC2(CO)CC2(C)C)CC1 CCC(C)(C)CC(=O)NCC1(C(N2CCC(CCCO)C2)=O)CC12CCC2 c1(CC(=O)NCCNC(C2(CC#C)CCCO2)=O)ccc2c(c1)CCCS2(=O)=O Cc1cc(C(N2CCCCC2C2CCN(C(C3(Cl)CC3)=O)C2)=O)c2n[nH]cc2c1 C(=O)(C(S(C)(=O)=O)C1CC1)N(CC(C)CNC(=O)C=CCOC1CCOCC1)C C1(C)(C(N2CCC(O)(CN(C(=O)CCS(C)(=O)=O)C)C2)=O)CC(O)CN1C C1(NC(C#CCNC(C(CCN(C)C)O)=O)=O)CC2(C1)CC(C#N)C2 c1(OCC=C)ccccc1CN1CCC(C(=O)Nc2cccc(Br)n2)CC1 C(=O)(C(C(C)(C)C)NC(c1ccc(CO)nc1)=O)N1C(CCC(C)C)CCC1 CCC1=C(C(=O)NCC2CN(C(c3cn(CCOC)nc3C)=O)C2)CCCO1 C(=O)(C1=NN(c2cccc(F)c2)C(=O)CC1)N(C(c1ccc(OC)c(Cl)c1)C)C c1(CC(=O)N(C2CCN(C(c3ncsc3C)=O)C2)CCC)ccc2ncsc2c1 CCCC(C(=O)N1CC2CCC1CN2c1ncnc(Cl)c1C)C(C)C c1(C(=O)NCC(C)(O)CNC(=O)CN2CCCCC2=O)cc(C2CC2)ccn1 N1(C(c2cnc(C)nc2C2CC2)=O)CCCC2C1CCN2C(=O)C=C1CCCC1 C1(N2CCN(CC(C)(C)S(C)(=O)=O)CC2)CCc2ccccc2C1 S(=O)(=O)(c1ccc(NC2CCSC(C)(C)C2)cc1Br)N1CC(OC)C(C)(C)C1 C1(CNC(CN(C)CC)=O)CC2(CCN(C(C3CC4(C3)CC(F)C4)=O)C2)CO1 c1(OC)cc(C)cc(C(C)NC(CCC(C)OC)c2nnnn2C(C)(C)C)c1F c1(OCC)ccnc(C(=O)NCCNC(C2CC2c2ccc(Br)o2)=O)c1 CN1C(=O)COc2ccc(-c3nc(C4(C)CCCO4)no3)cc21 C1(CN(C(NCC2C(C)C2)=NCc2ccc(F)cc2)C)Cc2ccccc2C1 CCC(C)C(C(=O)NCC(C)(C)NC(C1C(F)(F)C12CC2)=O)NC(=O)OC O=C(CS(=O)(=O)Cc1ccccn1)NC1CCCN(C(=O)Nc2cn[nH]c2)CC1 C1(NCc2ncc(C)o2)CCCC(CC(=O)NCCNC(CC(=O)OC)=O)C1 C1(CN(C(=O)Cc2ccn(C)n2)C)CCCCC1NC(=O)CSCC(N)=O c1(C(=O)NCCN(C2CCCC2)C(C2CCC(C)S2)=O)ccn2cnnc2c1 N(C(=NCC1CCCNC1=O)NC1CCOCC1)Cc1onc(CC)n1 c1(SC)ccnc(F)c1C(CN(CC(Cl)Cl)CC)=O C1(NC(CCSc2nc(C)[nH]n2)=O)CCCN(C(=O)Cn2cnnc2O)C1 N1(C(COCc2onc(CC)n2)=O)CC(NC(c2cncc(C)n2)=O)C(O)C1 C(=O)(C1=NOC(C)C1)NC(CC1CN(CC(=O)Nc2c(C)sc(Cl)n2)C1)C C=CC(C)CC(=O)NCC1CCCC(CNC(=O)CCSCc2ccccc2)C1 C=CCC(CC)C(=O)NCC1C(C(=O)NCC2(COCC)CC2)C1 N1(C(c2c(CC)cccc2CC)=O)CCC2CC1CN2C(=O)CCOCC(C)C N=c1[nH]c2ncc(C(N3CC4CCCC4(NC(=O)CC4(CO)CC4)C3)=O)cc2s1 c1(C(=O)NCCC(=C)CNC(C2(OC)CCCC2)=O)onc2ccccc12 C(=O)(C(C(C)(C)C)NC(=O)C(C)S(C)(=O)=O)N1CC(CC)(CO)C1 C(=O)(C(C(C)(C)C)NC(C1CCCN(CC)C1)=O)NC1CC(SC)C1.C(C)(C)(C)O C1(NC(COCCCC)=O)CN(C(C2CCC3CC23)=O)C2(CCC2)C1 Cc1nc(C(C2CCOC2)NCC(=O)OC(C)C)nc2c1CCCC2 c1(C(N(CC(C)NC(Cc2nc(C)sc2)=O)C)=O)cc(S(N)(=O)=O)sc1C C(=O)(CC1=CCN(C)CC1)NC(CCCC)CC(=O)N1CCN(C)CC(C)C1 CC1CCS(=O)CCN1C(=O)Cn1cc(CC2CCC=CCC2)nn1 C=CCCC(CC(C)C)C(=O)N1CCC(OCCNC(=O)C(CC)(CC)CC)C1 C(=O)(C(C)CC(=O)c1ccccc1F)N1CCCC(c2c(NCC)cccc2)C1 c1(C(=O)NC(C(C)NC(c2ccc(CC)cc2)=O)CO)cc(C)cc2c1OCC2 C#Cc1ccc(C(N2CCC(F)(CNC(=O)C(C)NC=O)CC2)=O)cc1C CC1CN(C(=O)Cc2cncc(O)c2)CC1CC(N1CCOCC1C(C)O)=O c1(C(=O)NCCOC2CN(C(C(C3CCOC3)OC)=O)C2)ccc(Cl)o1 c1(C(N2C(C)CN(C(=O)C(O)Cc3cn(C)cn3)CC2)=O)cc(N)c(F)cc1Cl N1(C(c2c(C)ccc(Cl)c2)=O)CCCC2(NC(C3CC3C)=O)CCCC12 N1(C(C(CC=C)(C)C)=O)CCC(NC(=O)CCC(C)(CC)CC)C(C)C1 C1(CNC(C(C)(C)N2CC=CC2)=O)CC(F)CN1C(=O)COCC(F)(F)F c1(C(=O)NCC2(OC)CCN(C(C3C=CCC3)=O)C2)ccc(C)c2ccccc12 C(=O)(CS(=O)(=O)C1CC1)N1CCCC(NC(C2CCC(N(C)C)C2)=O)(CO)C1 CCC(CC(=O)NC(CC(=O)N(C)CCc1cnn(C)c1)C1CC1)SC CC1CC(C(=O)NCC2(C)CSC2)CN(C(c2nnc(S)n2C)=O)C1 c1(OCC(=O)N(CCNC(C2CC(Cl)(Cl)C2)=O)CC)ccccc1Br S(=O)(=O)(c1cc(C)cnc1NCC1(CO)CC2CCC1CC2)NCC(CSC)C C1(C(N2CC(O)(CCNC(C=C(CC)C)=O)C2)=O)CC2C=CC1C2 C(=O)(C1=Cc2c(Cl)cccc2OC1)NC(C)CNC(=O)C(O)C1CCCC1 c1(C(=O)NC(C2(C(N3CCC(C)(O)CC3)=O)CC2)C2CC2)cnc2ccccn12 CC(C)(CO)C(=O)NC1CC(NC(C2CCNC2c2ccccc2)=O)C1 n1(N(CC(=O)N(CCC)C)CC(C)C)nccc1-c1ccccc1 c1(OCC)cc(C(=O)NCC2(C(=O)NCC3=CCCC3)CCC2)on1 c1(CC(=O)NCCC2(NC(C3C(C(C)(C)C)CC3)=O)CC2)c[nH]c2cnccc12 CCCC(CCNC(C1(CC)CCN(C(=O)CCCSC)CC1)=O)CCC C(CCC(=O)N(C)CCSC)N(C(C1CC(=C)C1)=O)C C1(NC(c2c(CC)scc2)=O)CN(C(=O)C(c2ccc(F)c(F)c2)O)CC12CC2 c1(C(=O)NC(CC)CN(C(=O)C(O)CF)CC)ccc2c[nH]nc2n1 CC12COCC1CN(C(=O)CONC(c1cncc(F)c1)=O)C2 N1(C(C(CC)(C)O)=O)CCC(C(N)=O)(Nc2nccc(C(F)(F)F)n2)CC1 C1(C(N2CCC(OCCCC)C2)=O)CN(C(=O)CC2CC(C)=NO2)CC(C)(C)C1 C1(CC)CCN(C(=O)CC2C=CC(NC(=O)CNc3cccc(O)c3)C2)C1C c1(C(=O)NC2(CO)CN(C(CCCNC(=O)OC)=O)C2)cc(I)ccc1Cl N1(C(C(C)OCC(C)C)=O)CC2CC1CN(C(=O)Cc1noc3ccccc13)C2 C1(N=[N+]=[N-])(C(N(C2CCCC2O)CC)=O)CCN(C(c2nnsc2N)=O)C1 c1(C(N2CCN(C(c3cc(Cl)ns3)=O)C3CC23)=O)ccn2ccnc2c1 COC1CCOc2c(C(N3CCC(N4CCCCC4=O)C3)=O)cccc21 N1(C(=O)C(O)c2cnc[nH]2)CCCN(C(C2(N3CCOCC3)CCCC2)=O)CC1 C1(C)(CNC(COC(CC)=O)=O)CCCN1C(=O)CCOCC(F)F C(=O)(CCC(C)CN(C)C)NCC(C(N1CCC(C)(N(C)C)C1)=O)OC N1(C(c2nocc2Br)=O)CCC2(CC1)CN(C(=O)C=Cc1ccc[nH]1)C2 C1(C(=O)NCCOCCNC(C2CC(COC)C2)=O)CCC1(F)F Cc1nsc(N)c1C(N1CC=CC(C(=O)NOC2CCN(C)CC2)C1)=O C1(C2CCN(C)CC2)(NC(c2cn(-c3c(C)cccc3)nc2)=O)CC1 n1(CC)ccc(C(=O)NCC2(NC(c3cc(C(F)F)no3)=O)CCOC2)n1 C1(C(N(CCNC(CSCC(C)C)=O)Cc2ccco2)=O)CCN(C)C1=O CC1CCn2ncc(C(N3CCN(C(c4cnccc4Cl)=O)C(CF)C3)=O)c2C1 C1(NC(C(C)CC2CC2)=O)CC2(C1)CC(NC(=O)C(c1cccnc1F)(C)C)C2 N1(C(C2(C(C)(C)C)CCCC2)=O)CCC(CCN(CCOCC)C)CC1 N1(C(C(C2CCCC2)NC(C(C)NC=O)=O)=O)CCCN(C)C(=O)C1 C1(C(N(CC(=O)NC2CC2)C)=O)CCCCCC1NC(=O)C1=CCSC1 n1(CC(=O)OC)c(C)cc(C(=O)N(CCCNC(C2COCCO2)=O)C)c1C N#Cc1cc(S(=O)(=O)NCC2CCCCC2)ccc1NCc1c[nH]c(=N)s1 N1(C(CCC(C)O)=O)CC2(CCOCC2)CC1CNC(=O)CCC(C)N(C)C N1(C(C2CN(C)C2)=O)CCCC(N(C(C2CCCC(=O)N2)=O)CC2CC2)C1 CC1CN(C(=O)NCC(F)(F)CN2CCOCC2)C(C)CCO1 C1(NC(c2c(COC)ncs2)=O)CC(F)(F)CC1NC(c1cncc(O)c1)=O CCCC(C(O)C(=O)N1CC(N(C)C)C(C)C1)NC(=O)Cc1ccc(C)o1 C1(NC(C(=O)NCCCN(OC)C)=O)CCCCC1N=[N+]=[N-] N1(C(C(N2C(c3cccc(OC)c3)CCC2)=O)=O)CC2(CC=CC(O)C2)C1 c1(NC(=O)OCC)ccc(NC(=O)CCc2csc(C)n2)cc1.C12CC(C1)NC2 [N-]=[N+]=NCCCCCC(=O)NC(C1CC=CCC1)C(=O)NCC1CC1Cl CC1=NOC(COC(C2(C)N(CCC(=O)Nc3ccc(C)o3)CC2)=O)C1 N1(C(C(CCOC)NC(c2ccc(OC)cc2)=O)=O)CC(F)CC(F)C1 C1(NC(CC(C)C)=O)CN(C(C)C(=O)NCc2cc(Cl)ccn2)CC1O C1(C(=O)N(C)CCN(C)C(c2cc(N)ccc2F)=O)(OC)CCC12CCC2 C1(C(C)C)CN(C(=O)C=CC2CC2)CCN1C(c1ccc(N)cc1O)=O N1(C(C=Cc2c(C)cccn2)=O)CCCN(C(=O)CC2CCOCC2)C(C)C1 N1(C(=O)OC(C)(C)C)CCC2(CCC2OC(c2nc(C(F)F)cc(C)n2)=O)CC1 C(=O)(CCCC(=O)N1CCOC(C(=O)NCCN(C)CCF)CC1)NCCC c1(CC)cnc(O)c(C(N2CC(NC(=O)CC3CCOC3(C)C)C3(CC3)C2)=O)c1 N1(C(Cc2c(C)ccs2)=O)CCCCC1CCN(C(=O)CN(C)C(=O)C1CC1)C N1(C(C(CC)OC)=O)CC(O)(C2(CNC(=O)C(C)CO)CC2)C1 C1(NC(c2csnn2)=O)CC2CN(C(=O)C(c3ccc(Cl)nc3)(F)F)CC2C1 c1(OC)ccc(CNC(c2conc2CNC(C2CC2C#N)=O)=O)nc1 C1(NC(C=NOC)=O)CC(C)CN(C(=O)CCc2csc(=N)[nH]2)C1 CC1(C)CN(c2nnc(CC3CCC(=O)N3)n2CC2CC2)CC(CCO)O1 C1(C(N2C(CCOC)CCCC2)=O)CCC2(CC2)N1C(c1ccc(=O)n(C)n1)=O c1(C(=O)NC(C(C)NC(c2c(C)cc(C)[nH]2)=O)C)c(C)nn2c(C)cc(C)nc12 c1(CC)cnccc1CNC(c1conc1NC(=O)CC1(NC(C)=O)CC1)=O n1(CCC(=O)OCCOCC#C)cnc2c(N)ncnc12 O=C(CCC1=CCCCC1)NCC1CC2CCC(C1)N2C(=O)CN1CCCCC1 C#CCCC(O)C(=O)OC.C12CCCN1C(=O)C2c1ccccc1 C=CCCCCCC(=O)NC12COC(C1)C(NC(=O)C(O)c1ccsc1)C2 C12(C(=O)OCC)CC3CC(CC(NC(=O)Cc4ccc(C)c(Br)c4)(C3)C1)C2 C1(C(=O)NCC(C)NC(c2ccc(CF)cc2)=O)CSc2ccccc2O1 Cc1c(C(N2CCCCC2CCN(C)C(C2CC2CN(C)C)=O)=O)cnn1C c1(C(N2CCC(N(c3ccc(I)cc3CO)C)CC2)=O)cc(C#N)ccc1Cl c1(CNC(c2cc(C)n(-n3cncn3)c2C)=O)cc2c(s1)CCCC2 C1(NC(CC2N(C)CCCC2)=O)CN(C(c2c(O)cccc2Cl)=O)CCC1(C)C C12(C(=O)NCC3OCC(CNC(=O)CCc4cncs4)C3)CCC(CC1)OC2 O=C1CCCC(CCC(=O)N2CC(CNC(c3csc(Cl)c3)=O)C2)N1 Cc1ccc(COCSCC(C(=O)NC(C)(C)C(C)CC(=O)OC(C)(C)C)O)cc1 CCC(C)CCCC(=O)N(C1CC(C(N2CC3CCC3(CO)C2)=O)C1)C C1(C(=O)NCCC(C)NC(=O)CSCCC(F)(F)F)OCCOC12CCC2 O=C(C1=CS(=O)CCC1)NCC1CCCCC1NC(C1(CCO)CC1)=O N1(C(C(CC)O)=O)CCc2c(C(=O)NCc3cnc(C(F)(F)F)nc3)n[nH]c2C1 C=CC(CCC)CC(=O)NC1CCCN(C(c2cc(-n3cnnc3)ccn2)=O)C1 c1(NC(C2N(C(c3c(C)cc(C)o3)=O)C(C)C2)=O)ccc2nc[nH]c2c1 C1(C2CCN(C(=O)Cc3cn4c(n3)CCCC4)C2)(NC(C2N=C(C)SC2)=O)CC1 c1(C(N(C2CN(C(c3cc(C)c(C)s3)=O)CC2O)C)=O)coc2c(C)cccc12 N1(C(C(C)N2CCC2)=O)CCCC(C2CN(C(=O)Cc3ccc(Cl)cc3)C2)C1 C12N(CC1(C)C)C2=O.C1(CC(=O)NC2C=CC(COC)C2)CC2(CC2)CO1 C(=O)(CN=c1ccc(Cl)n[nH]1)NC1CC(N(C(=O)CC2CN3CCC2CC3)C)C1 CN1CCC(N(C)CC2CCN(C(c3ccccc3C(F)F)=O)CC2)C1=O N(C1COc2ccccc21)C(C(CCF)NC(CCNC(C)=O)=O)=O C1(C(=O)NCC(C)(CO)NC(Cc2c(CC)cccc2)=O)CCOCC1(C)C N1(C(C=C(C)C(C)(C)C)=O)CCC(NC(c2ncccc2C)=O)C12CCC2 C1(OCCOC)CC2CN(C(c3ccc(OCCn4ccnc4)cc3)=O)CC12 C1(CC(N2CC(O)(CNC(COCC(N3CCCC3)C)=O)C2)=O)CCCC(O)C1 N1(C(C)=O)CCC2OCCN(C(c3ncn4cc(-c5ccnn5C)sc34)=O)C2C1 C=CCCCCCCC(=O)NC1CC2(C1)CN(C(C1CCCCN1C)=O)C2 Cc1nccnc1C(=O)NC1CC(C)N(C(=O)CCCN2CCCC2)C1 N1(C(CCCN(C)C)=O)CCSCC1CN(C(C1CCC1F)=O)Cc1ccccc1 Cc1cscc1C(=O)NCc1occc1C(=O)NCC1CCOC1C(C)C c1(NC(C)C(=O)NCc2ccc(C(=O)N(C)CCOC3CC3)o2)ccc(F)cc1 N1(C(c2nc(C)sc2)C(=O)NN2CCCC(N3CCOCC3)C2)CCCC(C#N)C1 c1(CCC(=O)NCC=CCNC(C(C)CC2CCC2)=O)nc2ccccc2o1 c1(C(=O)NCCCC(C)NC(c2c(C)coc2C)=O)coc2c(Cl)cccc12 C(CC(C)C(=O)NCc1ccc(C(=O)NC2CC(=O)N(C)C2)cc1)=CC N1(C(c2ccc(C(c3ccccc3)=O)o2)=O)CCCC(O)C1C(F)(F)F CC1C(C)N(C(C23CC4CC2C3C4O)=O)CCN1C(c1ccc2occc2n1)=O C(=O)(C(C)(C)C)NC(C1CCCN1C(=O)Nc1ccc(CN2CCCC2)o1)C CCCCC(C)(F)C(=O)NC1CCC(NCc2cccc3scnc23)C1 C1(NC(=O)NC2CC(N3CCOCC3)C2)CCC2CCCCC2C1 C(=O)(C(C(=O)N(CC(C)NC(c1cc(F)ccc1CC)=O)C)C(C)C)OCC c1(OC)ccc2nc(N3CC=CC(NC(=O)C(C)NC(=O)CC#N)C3)sc2c1 Brc1cc2c(N3C4CN(Cc5cccc(-n6cncn6)c5)CC34)ncnn2c1 c1(C(=O)Nc2c(NCC)ccc(Cl)c2)ncc2ccccc2c1O C(=O)(C1CCCc2nncn21)N1CC2(OCC(NC(=O)COc3cn[nH]c3)C2)C1 C1(C2(O)CCOCC2)(C(N2CC(CNC(C(CC)=CC)=O)C(C)(C)C2)=O)CC1 C#CCCCCC(=O)N1CCCC(C)(C(=O)NCC(C)(F)F)C1 c1(OCC(=O)NC2(C#C)CC2)ccc2c(c1)CCCC2=O.C1CS1 c1(NC(C2N(S(CC)(=O)=O)CCSC2)=O)ccc2c(c1)n(C)c(=O)n2C CC12CC(N(C(C3CN4CCCCC4CO3)=O)C3CC3)(C1)C1(CN(C(=O)CO)C1)O2 C1(NC(c2c(C)nn(C(C)C)c2)=O)CN(C(=O)CO)C(C)(CN(C)C)C1 C(=O)(CS(=O)(=O)CCOC)NC1C=CC(C(=O)NC(CCCC)CO)C1 Cc1cc(C(=O)NC(CO)CCCNC(c2cc(F)c[nH]2)=O)nn1C(C)C1CC1 C1(C(=O)NCCCCN(C(=O)C(c2cscn2)N(C)C)C)CC12CCSCC2 N1(C(C(CCNC(=O)OC(C)(C)C)(C)C)=O)CCC(C2=NOC(C(=O)O)C2)CC1 c1(N(CC(=O)NC2CCC3(CCNC3)OC2)C)nc2ccc(N(C)C)cc2[nH]1 CC(C)CC(=O)NCC(N1CCC1CNC(C1CC(C(F)F)C1)=O)=O CC(C)C(C(=O)NC1CC1NC(C1CC(n2ccnc2)C1)=O)NC(=O)C1CC1 C1(C(=O)OC)CCN(C(=O)C2CC2c2cncn2C)O1 C(=O)(CC(CC)NC(=O)Cn1cc(C#N)cn1)NCC(=O)NCC c1(C(N(C2CC(NC(=O)COC(C3CCC3)=O)C2)C)=O)ccc(C2CC2)c(F)c1 C(CCSCC)(C(=O)Nc1nccc(C(F)(F)F)n1)N(CCCOCC)C N1(C(Cc2nc(C)cc(C)n2)=O)CCC2(CCN2)CC1 C(C(=O)NCC1CCCCN1C(=O)COCCOCCO)(C(C)C)OC C(c1cc(C)c(C)cc1C)=CC(N1CCN(C(C2(C#C)CC2)=O)CC(O)C1)=O C1(C(N2C(C)C(C(=O)NCCCCCCF)CC2)=O)CCCCC1(C)C c1(CC)ccc(C(=O)N(C(C)CNC(=O)CCCN(C)C)C)cn1 Cc1cc(=NC(=O)C(=O)N(C(c2ccc(F)cc2)CC2CN(C(C)=O)C2)CC)[nH]o1 c1(OC)cnnc(C(=O)NCC2(NC(=O)C(c3ccccc3)C)CCOCC2)c1 c1(C(N(C)CC2(O)CN(C(=O)CCS(C)=O)C2)=O)ncncc1Br c1(OC)ccc(N(CC(C)O)Cc2cccc(C3COC3)c2)cc1 C1(N(C(=O)CC2CC3CC3C2)C)CCCN(C(=O)CSCc2cccs2)C1 c1(C(=O)NC2CC(NC(Cc3cc(C(C)C)no3)=O)CC2O)c(Cl)cncc1Cl C(CCCCC(=O)N1CCCN(C2CC2)CC1)NC(c1cc(OCC)n[nH]1)=O C1(C(N(CCNC(COCC(=O)NC)=O)C(C)C)=O)CSCC(=O)N1 CC1CCCn2ncc(N(C3CCCCC3)C(C3CCN3C(=O)OC(C)(C)C)=O)c21 C1(C(N2CCC(CC)(CO)C2)=O)CCN(C(c2ccoc2C2CC2)=O)C1(C)C N1(C(CSCC#C)=O)CCCC(C2CCCN2C(=O)C=CC(c2ccsc2)=O)C1 CC1CNCCC1NC(C1(CC2CC2)CNC1)=O c1(C(=O)NCCc2ccc(C(N)=O)cc2)occ2c1CCC2 C1(CNC(c2c(C)cncc2)=O)CN(C(c2coc(Cl)n2)=O)CC12CC2 c1(C(N2C(C(N(C3CCOCC3)C)=O)CSCC2)=O)cc(O)nc(O)n1 c1(OC)nc(Cl)cnc1NC(C1CCCN1C(c1cccc(F)c1SC)=O)=O c1(C(N(C2CCN(C(C3CN(C(=O)N(C)C)C3)=O)CC2)CC)=O)nccnc1N C1(NC(n2c(C)csc2=O)=O)CC(NCC(N)=O)C12CCC2 CCCCC(C(=O)NC1CC=C(C)CC1)NC(c1cc(Cl)cn1C)=O C(=O)(CC(O)c1cnc(Cl)s1)NC1(CNC(CC2CC(OC)C2)=O)CCC1 N(C(=NCCCOCC1CCCC1)N1CCC(C(C)OC)C1)CCOCC N1(C(C2(C)CCCO2)=O)CC2CN(C(C34CC(CCO3)C4)=O)CC2(C)C1 C1(CC(N2CCCC2(C)C2CCC2)=O)C2CCCC2N1C(C1(F)CC1)=O.CC=O c1(C(=O)NC(C2CN(C(=O)C3=NNC(=O)CC3)C2)C)cc2c(F)ccc(F)c2s1 c1(C(N2C(CCNC(C(COC)C)=O)CSCC2)=O)cc2cc(C)ccc2[nH]1 C1(CC#C)(C(N2CCC(O)(CNC(=O)C(C(C)C)NC(C)=O)C2)=O)CC=CCC1 c1(C(N2CC(C)C(NC(=O)CC3CC3(Cl)Cl)C2)=O)ccc(N)c(F)c1F Cc1cc(-n2cccc2)ccc1C(=O)N(C1CN(C(c2c[nH]c(=N)o2)=O)C1)C c1(C(N2CC(F)CC(C(N3CCCC(CO)C3)=O)C2)=O)cccc([N+](=O)[O-])c1I C=CCC(CCCCC)C(=O)N1CC(CN)C(C)(C(C)C)C1 CCCC(CNC(C1COCC(C)O1)=O)C(=O)N1CCC(C#N)C1 C12(C(N3CCC(C)(CNC(COC)=O)C3)=O)CCOC1CCOC2 c1(OCC(=O)NCC2(NC(c3csc(CO)n3)=O)CC2)ccc(F)c(F)c1 Cc1sc(C2CCCN(S(=O)(=O)CC34CC(C)(CO3)C4)C2)nc1C(=O)O C(=O)(CC(O)CNC(c1cccn1C(C)C)=O)NC(C#C)(C)C N1(C(C2CN(C(C)=O)C2)=O)CC2CC1CCN2C(c1cccc([N+](=O)[O-])c1)=O CCC(C)C(C)CNC(c1cn(CCNC(=O)Cc2cc[nH]n2)cn1)=O c1(C(=O)NCC2C(NC(C(CC)OCC)=O)CCC2)cn2cccc(F)c2n1 c1(C(=O)NC2CCCN(C(c3ccc(SC)cc3)=O)C2)cc(S(C)(=O)=O)cs1 C1(C)(C(=O)NCCCOC)CC(O)CN1C(=O)C1=COCC1 c1(C(N(CCNC(CCCCC=C)=O)C)=O)cc([N+](=O)[O-])ccc1NC(=O)OC C12(Nc3c(C)cncn3)CCCCC1CN(C(C1CC1C)=O)C2 C=CCC(CC)C(=O)N1CCC(C)(CC(N2CCCC(C(C)(C)C)C2)=O)C1 N1(C(C2C(CC)C2)=O)CC(NC(C23CCC(C)(CC2)CO3)=O)CC12CCCOC2 N1(CCCCC#C)CC2CN(C(c3cccc(CCC)c3)=O)C2C1 C(C)(CCC(=O)NCC1CN(C(C2CC(F)C(=O)N2)=O)CCO1)OC c1(OC)nc(C)ccc1C(=O)NC1CC2CC1N(C(=O)C1=CCSC1)C2 CC1=C(C(=O)NC2(C)CCC(NC(=O)CC3CCC3(C)C)CC2)CCCC1 c1(-c2cc(CN3CCN(S(C)(=O)=O)CC3)[nH]n2)cccc(F)c1F Cc1cc(CC(C)NC(c2[nH]ccc2CNC(=O)Cn2nccn2)=O)n[nH]1 C1(N(C(C(CC2CC2)OC)=O)C)CCC(NC(=O)C(C)(C)CO)CC1 C1(C(=O)NCC(CNC(CC2(CC)CC2)=O)(C)O)CC(=O)N(C2CCCCC2)C1 N1(C(C2C(C)(C)C2)=O)CCC(C)(C)C1C(=O)Nc1cnccc1CO C12(C(=O)NC(CC)CNC(C3CC34CCC4)=O)CCC(OC)(CC1)C2 Cc1ccc(CN2C(C(=O)Nc3cccnc3CO)CC3CC23)cc1Br N1(C(c2cc(CCC)on2)=O)CC2CC(NC(=O)C(C3CCCCC3)C)CC1C2 C1(C(N(CCCCNC(c2cc(C)nn2C)=O)C)=O)CC(C)CCC1C(C)C c1(C(=O)NC(CCCC)C(=O)NC2(CO)CC(F)C2)ccc2c(c1)OCO2 C(=O)(C(C)C(F)(F)F)NCC1(NC(C(c2ccc(C)cc2)C2CCC2)=O)CCC1 CCCC(C)(C)C(=O)NCC1(C(C)(C)C)CCN(C(c2c(C)cc[nH]c2=N)=O)C1 c1(C(N2CC(SC)C(NC(=O)Cc3cc(Cl)n(C)n3)C2)=O)cnc2ccnn2c1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC2(CC(NC(CC(C)OC)=O)C2)CC1 C(C(C)(C)CC(=O)NCC1(CC2CCC2)CC1)NC(C(C)CN(C)C)=O c1(C(=O)NC(C)C(CO)NC(=O)CCc2cccs2)cc2n(n1)CCC2 C1(C(=O)NC(C2(O)CN(C(CC3(C=C)CC3)=O)C2)C)CCCN(c2nccs2)C1 C(C1=NOC2(CCC2)C1)CNC(=O)NCc1nnc(-c2cc(Cl)ccc2F)o1 c1(C(N2CCC(C)(NC(C3CC34CCCCC4)=O)C2)=O)ccc2ncnn2n1 C1(C(=O)NC2(CO)CCOC2)C2CCC1(c1ccc(C(F)(F)F)cc1)C2 C1(C(=O)NCC2CC(NC(CC(CC)C(C)C)=O)C2)CCc2ncncc2C1 N1(C(C2C(CC)OCC2)=O)CC2CCC1C1CN(C(=O)C(C)(C)CF)CC21 c1(OC)ccc(OC)c(C(F)(F)C(=O)NCC(C)NC(C2CC2(C)C)=O)c1 Cc1c(Br)ccc(C(=O)NCC(c2ccc(Cl)s2)O)c1F C(=O)(C(C)CC(N)=O)NC(C)C(=O)NCC1(O)CN(C)C1 N1(CC2N(C(C3CCCCO3)=O)CCCC2)CCCCC(n2cc(CO)nn2)C1 c1(N(C(C2CCN(CCC)CC2)=O)CC)ccc2c(c1)C(C1CCNCC1)C(=O)N2 c1(C(N(CC(CC)NC(c2ncncc2F)=O)CC)=O)cccc2cncn12 CC1CC=C(C(=O)NC2CCN(C(C3COC(=O)C3)=O)C23CCC3)CC1 c1(C(=O)NC2CN(C(CCC3N(C)CCC3)=O)CC2O)cn2cccc(Cl)c2n1 n1(CCC)cc(Cl)c(C(N2CC(NC(c3cscc3C(N)=O)=O)C(C)C2)=O)n1 N1(C(c2c(CC)con2)=O)CC(C)(C)CC1C(=O)NCCc1cc(C)[nH]n1 CC(O)C(CNC(=O)COCC1CCCC1)NC(=O)CCc1cncs1 c1(CC)ccc(C(C)NC(=O)CCc2cccn2C)cc1 c1(CC(=O)NC2(CO)CCCN(C(C3CC34CC4)=O)C2)c[nH]c2ccccc12 CC1(C)CCCCC1CC(=O)N(CCNC(c1cc(C(N)=O)[nH]n1)=O)C1CC1 C(=O)(C(C)(C)C(C)(C)O)N1CC(O)(C(C)NC(C2CCCC(O)C2)=O)C1 N1(C(c2cc(C(C)C)no2)=O)CCOCC1C(=O)NCCC(C1CC1)C1CC1 CN=S1(=O)CCN(C(C(=O)NCc2ccc(F)cc2)C2=CCSC2)CC1 CC(C)CC(C(=O)NC1CC(C(=O)N(CCCN=[N+]=[N-])C)CC1O)C(C)C N1(C(c2c(C)cc(C)s2)=O)CC2CCC1C(NC(c1cnn(CCF)c1)=O)C2 C1(COC)CC(O)CN1C(=O)CN(C(c1snnc1C)=O)C1CC1 c1(N(CCCCCC)C)ccc(S(=O)(=O)NC2CC(NC(C)CO)C2)c(Cl)c1 N1(C(c2cc(CC)on2)=O)CCCC(CC(=O)NC(C)CCn2cncn2)C1 C(=O)(C(O)CC(F)(F)F)N(c1cnn(C)c1)CC(N1CCC(OC)C(C)(C)C1)=O c1(CCCC)ccccc1OCc1ccc(Cl)cn1 C1(NC(c2c(C)nc(Br)o2)=O)CC(C)CN(C(c2cn(C)nc2C(F)F)=O)C1 C1(NC(c2c(C)ccs2)=O)CCCCC1CNc1ccnc(CO)n1 c1(CC(=O)NC(CNC(C(C2CCC2)OC)=O)C)coc2c(Cl)c(Cl)ccc12 Cc1cn(C)cc1C(=O)NC1CC(NC(C2CCCC3CC23)=O)C1 C1(NC(c2cccc(C)c2F)=O)CC12CCN(C(c1cnc(O)cc1O)=O)CC2 CCC(C)C(C(=O)N1CCC(CCc2nccc(C(C)(C)C)n2)C1)N(C)C N1(CC(=O)NC2(C(N3C(CC(=O)NC)CC3)=O)CC2C)CCCCC1C C1(Nc2c(OCc3ccncc3)ccc(F)c2)C2CCc3ccccc3C12 Cc1nc2cc(C(=O)NC34CCCC3CN(C(C3(N(C)C)CC3)=O)C4)ccc2s1 NC1CCC(F)(F)CC1C(=O)NCC1CCCCN1CC(F)F Cc1nn(C)c(Cl)c1-c1cn(C2CN(C(C3CC4CC3CC4=O)=O)C2)nn1 c1(OC)ccc2oc(C(=O)N(CC(c3nn[nH]n3)C)CCO)cc2c1 Cc1cc(C)c(C(N2CCC(=CCNC(C3C4CC4C4CC34)=O)CC2)=O)c(O)c1 Cc1cc(C(N2CCC(CNC(=O)C3=C(Cl)CCOC3)C2)=O)n2ncnc2n1 c1(C(N(C2CCN(C(c3cc(C)c(C)o3)=O)C2)CCO)=O)ncc2ccccn12 c1(-n2cc(C(CC)O)nn2)cccc(CCNC(C2(C)CCCN2C)=O)c1 c1(C(N(C2CCCN(C(c3c(OC)csc3)=O)CC2)C)=O)cccc2ccnn12 C(=O)(CC(C)SC)N(C)CC1(C(=O)NC(C2CCCCC2)C#C)CC1 C(CNC(c1cnc(C2CC2)s1)=O)(CC(F)(F)F)NC(c1cccc(C)c1)=O.C1CC1 C1(CCNC2OCCC2(CC)C(=O)NCc2ncc(CC)o2)CC(=O)N(C)C1 Cc1ccc2c(c1)CC(C(N(CCc1nn[nH]n1)CC13CCC(CC1)C3)=O)S2 c1(C(N2CC(N(C(c3cc(C(C)=O)sc3)=O)C)C2)=O)cc(O)nc2c1CCCC2 c1(NCC2CCOC2)cccc(S(=O)(=O)Nc2c(Cl)nc(C)c(Br)c2)c1 C1(NC(COC(C)C)=O)CC2CC1N(C(=O)CC1CCCC(=O)C1)C2 c1(NC(C(=O)N(CCC#C)CC)=O)ccc(Oc2ccc(F)cc2)nc1 Cc1ccc(C(=O)NCC(C2CCCC2)OC)c(C2CC2)n1.C1(=O)CC(C)N1 CC1(CC#N)CCN(C(=O)C(=O)NCCC2CC2)C1 C12(CNC(CCCC)=O)CCCC1CCN2C(c1cccc(OC(C)C)n1)=O C(=O)(CCCCCCn1cnnn1)NC(CC)CNC(c1c(C)n[nH]c1C)=O C1(CNC(CC=CC=C)=O)CCCCN1C(=O)CC1(N(C)C)CC1 c1(C(=O)NC2CCC(N(C)C(c3cnccn3)=O)C2)cnc(O)c2c1NCCC2 C=Cc1cccc(CN2CCC2C(=O)Nc2ncccc2OC)c1 c1(C(N2CCCCC(NC(C(C)S(C)(=O)=O)=O)C2)=O)ccc([N+](=O)[O-])cc1O N1(C(c2cnccc2Cl)=O)CC2CC(C1)CN(Cc1c[nH]c3ccc(Cl)cc13)C2 CC1=NS(=O)(=O)NC(C)=C1CC(=O)NCCCNC(=O)C(C1CCC1)C1CCC1 Cn1cnc2c1CCC(C(=O)NC(CNC(=O)CSCC(N)=O)C(C)(C)C)C2 C1(CCNC(CCCCC)=O)CC2CCC(C1)N2C(c1c[nH]nc1C(F)(F)F)=O c1(N(CC(CN(C(C2(OC)CCCC2)=O)C)O)C)ncnc2scc(Br)c12 c1(CCNC(c2ccc(Cl)s2)C)ccc(F)c(Br)c1 Cc1ncc(CC(=O)N(CC(C)C#N)C2CC2)s1.C12CCC(C1)NC2=O S(=O)(=O)(C1CN(C(=O)CCC(N)=O)C1)N1CCN(C(CC2(COC)CC2)=O)CC1 Cc1ccc(O)c(C(N2CCC(NC(c3cn(C(C)C)nn3)=O)C(C)C2)=O)c1 CCC(O)C(=O)C1C(C(=O)NC2CC(NC(=O)C=CCOCCOCCOC)C2)C1 C1(CNC(CC(C)(C)O)=O)CN(C(c2cc3ncccc3s2)=O)C2CCN1C2 N1(C(=O)C=Cc2cccnc2)CCC2CN(C(=O)Cc3cccs3)CCC2C1 c1(NC(C)=O)ccc(O)c(NCCCO[Si](C)(C)C(C)(C)C)c1 C12(NC(c3c(C)nsc3)=O)CCOCC1CN(C(=O)CCc1ccc(Cl)nc1)C2 c1(C(=O)NC2CC(NC(C(C)SCCCC)=O)CC2O)nn(C)c(Cl)c1Cl C1(NC(c2cnc(C)nc2)=O)C(CNC(=O)Cc2ccc(C)s2)CCC12CCC2 C1(CN2CC3CN(Cc4cccc(OC)c4)CC3C2)COc2ccccc2O1 Cn1cccc1C(=O)C(=O)NCC1(C(=O)NCCCC2CCCO2)CCC1 Cc1ncncc1C(=O)NC(C(=O)N1CCC(C(F)F)C1)C(C)C Cc1cc(SCC(=O)NCCNC(C2(C(O)C#N)CC2)=O)cc(C)c1 CCCCC(C)(CO)NC(C1CCC(NC(c2nn(C)cc2C)=O)C1)=O C(=O)(C(C)CC(C)(F)F)N1CCC(CCN(C(CC(C(C)C)O)=O)C)CC1 c1(C(=O)NC(C2CCN(C(=O)C=C3CC3)CC2)CO)ccc(Cl)c(F)c1 C1(C(=O)NCC(C)N(CC)CC)CC(F)(F)CN1C(C1CC(=O)CC(=O)C1)=O c1(NC2(c3nc(C)cc(C)n3)CCCCC2C(C)(C)C)c(O)cc(F)cc1F Cc1[nH]nc(CO)c1C(=O)N(CC(C)C(=O)NC(C1CCC1)C1CCC1)C N#CC12CC(C(N3CCC(CCNC(=O)CSCc4ccccc4Cl)C3)=O)(C1)C2 c1(NC(C2CC2CNc2cnccc2-c2ccccc2)=O)nccn2ccnc12 N1(C(C23N(C(C(C4CCC4)OC)=O)CC(C)(C2)C3)=O)CCn2ccnc2C1 C1(C(=O)NCC(C)(CO)NC(=O)OC(C)(C)C)CC2(CCC2)CCO1 C(c1ccc(Cl)cc1)=CC(=O)NCC1N(C(c2nc(CCC)oc2)=O)CCC1 N1(C(C(CCC)(C)CCC)=O)CCCC2(CCCN2C(=O)C(O)P(C)(C)=O)C1 C1(NC(c2c(OC)nn(C)c2)=O)CCCN(C(c2cnc(N)cn2)=O)CC1 C(c1cccc(F)c1F)=CC(=O)NC1(C2CN(C(Cc3ccc(C)s3)=O)C2)CC1 C(CC(=O)NOCCCF)C1(C)CN(C(CC2(OC)CC2)=O)C1 Cc1occc1C(=O)NC(c1cccnc1)C(=O)NC(C1CCC1)C c1(C(=O)NCC2CN(C(C3C(CCC)C3)=O)C(C)(C)C2)n[nH]c(CC)c1[N+](=O)[O-] C1(CC(=O)NCC2CN(C(c3c(C)ocn3)=O)C(C)C2)CC(C)(C)OC(C)(C)C1 c1(-c2occ(C(=O)NCC(CC)NC(c3cnc(S)nc3)=O)n2)ccc(Cl)cc1 N1(N(C2CCS(=O)(=O)C2)C)CC(NC(=O)CC(C)(C)C)C(C)(C)C1.C=O N1(C(C2C(C(=O)NCC#C)C2)=O)CCC(NC(=O)COC(F)F)CC1 C1(CC)(CC)CC(NC(c2cc(Cl)no2)=O)CN1C(=O)Cn1cc(C)cn1 C(=O)(C(CC)C(=O)NC(C)CCNC(=O)CCc1ccc(C)nc1)OCC C(=O)(C(F)CC(CC)CC)NC1(CC=C)CCN(C(=O)CNC(=O)CN(C)C)C1 C(=O)(C1CCCc2scnc21)N1CCC2(CN(C(c3cccc(F)c3Cl)=O)C2)C1 C1(C(=O)NCCCCOCC)CN(C)CCN1C(c1cnccc1C#N)=O c1(CC(=O)NC2C(NC(c3c(OC)n[nH]c3)=O)CC2)cc(O)nc(O)n1 C(=O)(C#CC1CCCC1)NC(CC=CC)C(=O)NC1CCOCC1(C)C O=C(C#CC1CCOCC1)NCCC12CCC1CN(C(c1cnn[nH]1)=O)C2 C=CCCC(O)CN(C(=O)C(C)(CO)NC(c1cccc(F)c1)=O)C C1(F)(CNC(CC2(OC)CC2)=O)CCN(C(c2c(C)cc[nH]c2=N)=O)CC1 C1(C(=O)NC(C(=O)NC(c2onc(C)n2)CO)C2CCCC2)C2CCC(C2)C1C Cc1cc2ccc(C(=O)NC3CN(C(=O)CCc4nnc(C(C)C)o4)C3)cn2c1 C1(C(=O)NC(C)(C)C)CCCN(C2C=C(Br)CC2)C1 C1(N(C(=O)NCCCc2ccccc2)CC2CCSCC2)CCCCC1(F)F c1(C(=O)NC(CC)CNC(c2cccs2)=O)cc(Br)cc([N+](=O)[O-])c1 C1(NC(c2n(C)ccn2)=O)COCCN(C(c2snc(Cl)c2Cl)=O)C1 N1(CC)CCCCC1CN(CC(C)O)C(c1ccc(-n2cccc2)cc1)=O C1(CNC(C2C(C)C2C)=O)CN(C(=O)Cc2csc(C(N)=O)n2)CCC12CCC2 O=C(CCCC1CCCO1)N1CCCC1C(O)C(N1CCC(N2CC(O)C2)C1)=O N1(c2c(C(=O)OC)c(Cl)ncn2)CC2(CCCN2C(c2cscc2C)=O)C1 C1(CS(=O)(=O)N(CC(=O)OCC)CC)(Cc2ncc(Cl)s2)CC(F)(F)C1 C1(C(=O)NCCC2(CNC(CC(C)c3cccnc3)=O)CC2)C2CCC(F)(F)C12 CC1(C)CCCC(C(=O)NC(C(=O)NCC2(CO)CC2)C2CCCC2)C1 C#Cc1cn(C)nc1C(N1CC2CC(NC(c3cnccc3OC)=O)C1C2)=O C1(CN(C(=O)C(c2ncccc2F)(F)F)C)CCCN(C(=O)C(C)(C)C)C1 C1(C(N2CC(O)(C(=O)OC)C2)=O)CC(C)CN(C(c2ccc(O)cc2)=O)C1 N1(C(c2scc(C)c2)=O)CC(CNC(c2ccccc2-n2cccn2)=O)CC1C c1(C(N2CC(CC(C)NC(C3(C(C)(F)F)CC3)=O)C2)=O)ccc(N)c([N+](=O)[O-])c1 C1(CC)CN(C(c2csnc2Cl)=O)CCN1C(c1cnc(C)cc1C)=O C(c1cccc(F)c1)=CC(=O)NCCC(C)NC(C1(C)CCC1)=O c12cccc(c1)S2.C1(N(C)C(C2(CO)CC2)=O)CCCC(NC(=O)C(F)F)C1 C1(CNC(=O)CCc2cncnc2)CC2(CC(NC(C3CCCCO3)=O)C2)C1 CCC(CC)C(F)C(=O)NCC1CCCCCN1C(C1CCCC(CF)C1)=O N1(C(Cc2c(C)non2)=O)CCOCC(C(=O)NC(c2ccccn2)CO)C1 C(C(C(C)C)NC(c1cc(C2CCOCC2)[nH]n1)=O)NC(C1CC(C)C1)=O N1(C(=O)OC(C)C)CCCC1C(=O)NCCCN(C(=O)CC1CCSCC1)C C=C(C)CCC(=O)NCC1C2CC1N(C(c1oc(-c3ccccc3)nc1C)=O)C2 S(=O)(=O)(c1ccc(CNC)cc1)N(C(C(=O)OCCC)(C)C)S(C)(=O)=O CCCC(C)(CC)C(=O)NC1CCC1NC(c1coc(C2CCCCC2)n1)=O CC1CN(C(C2(N)CCC2)=O)C(C)C(C)(C)O1.C(=O)(C=CCO)N1CCC1 C1(NC(CNC(C(CC)C)=O)=O)C2CN(C=O)CC12.C1(C)(C2CC2)CCCO1 N1(C(=O)Cn2cc(C3CC3)nn2)CC2CCC(C1)N2C(=O)CCC1CC1(F)F c1(C(N(CC2N(C(C3C(COC)C3)=O)CCC2)CC)=O)cc(=O)c(OC)cn1C c1(NC(c2ncc(-c3ccc(CC)nc3)c(OC)c2)=O)cnccc1[N+](=O)[O-] c1(NC2CN(C(c3ccnn3C3CCCC3)=O)C2)ccc([N+](=O)[O-])cc1Cl CC(C)C(CNC(c1cnn[nH]1)=O)NC(=O)CSCc1ccccc1 C1(CC(=O)N(C(C)C(=O)NCC2(CC3CCC3)CC2)CCC)CC=CCN1C c1(C(N(CCC(C)NC(=O)CC(C)C(F)(F)F)C)=O)coc2cc(F)ccc12 c1(NC(c2c(CNC(C(C)OC(C)(C)C)=O)occ2)=O)ccc(CO)cc1 N1(C(=O)OC(C)(C)C)CCC(C)(C(=O)C(F)(F)F)C1.N1(C=O)CCN(C(=O)NCO)CC1 N1(C(c2c(C)nc[nH]2)=O)CC2CN(C(=O)CNC(c3cccnc3Cl)=O)CC2C1 C(=O)(C(C)(O)CC(F)(F)F)N(CCCC)CC(=O)NCCOC(F)F c1(C(=O)NC2CCN(C(c3ccc(C)cc3)=O)C2(C)C)snc2ccccc12 CN1CCCC(F)(C(=O)NC2CC(CCNC(C3CC(C)(C)CO3)=O)C2)C1 C1(C(=O)NC(C)CCc2ccc(F)cc2F)CCN(C(=O)C(N)=O)CC1(C)C C(=O)(C(C)(C)CS(C)(=O)=O)N(C1CCN(C(C2CCC(O)CC2)=O)CC1)C N1(Cc2c(OC)cccn2)CC2CCC(C1)C2NC(c1cc2cnccc2[nH]1)=O N1(C(CC2CC(=O)NCC2)=O)CCC2CN(C(=O)CCC3CCCO3)C2C1 c1(C(N(C2CCN(C(=O)CSC(C)C)CC2)CCC)=O)cn(C(F)F)c(C)n1 n1(CC)ccc(CC(=O)NCCNC(C=CCN(C)CC)=O)n1 CCC(C)(C(=O)N(CCCNC(c1cn(C)nc1C(C)C)=O)C)OC c1(C(N2CC(O)CC(NC(C3(OC(C)C)CCC3)=O)C2)=O)cc2cnn(C)c2s1 Cn1ccc2cc(-c3ccnc(NC(c4nc(Cl)cs4)=O)c3)cnc12 C1(C(=O)OCC)CCC(C(=O)NCC2COCC2NC(C2(C#N)CC2)=O)CC1 CCCC(CC)C(=O)N1CCCC(CC)(NC(=O)CC2(C#N)CCC2)C1 c1(C(N2CCC(O)(CNC(C3C(C)OC(C)C3)=O)CC2)=O)cc2ccccn2n1 c1(C(=O)OC)cc(I)c(N(C)Cc2c(OC)cnn2C)cc1Cl C1(C(C)NC(C2C(C(=O)OC)C2)=O)CN(c2ncc(C(F)F)cn2)CCCO1 c1(C(=O)NCc2c(OCCOC)nccc2)ccc2c(c1)ncn2C(C)C c1(C(=O)NCC(N(C(=O)CC2=NNC(=O)C2)C)OC)ccc2ccc(O)nc2c1 CC(C)(C(=O)N1CCC1(C)CC(=O)NC1C2CC(O)CC12)C(N)=O C1(NC(C(C)n2cncn2)=O)CC(F)(CNC(=O)C=CC(c2ccccc2)=O)C1 c1(NC(CNC(C(CC)CN(C)C)=O)=O)cnc(Cl)nc1C C12(NC(=O)CN3CC=CC3)CCC(CC1NC(=O)C(O)(C1CC1)C1CC1)C2 C1(CC(=O)NCCCCCCN(C)C(C2CCS(=O)(=O)C2)=O)CCCCC12CC2 c1(C(C(=O)NCC(C)N(C(c2cn(CC(C)C)nc2)=O)C)O)ccc(Cl)c(Cl)c1 c1(CS(C)(=O)=O)ccccc1C(=O)N(CCO)NCc1ncn(C)n1 Cc1c(C(N2CCCC2CNC(=O)CC(C)(C)O)=O)cccc1O N1(C(C2CNC(=O)N2)=O)CC2CC1CN(C(C1(c3ccc(F)cc3)CCC1)=O)C2 C1(CCNC(C2(SC)CCC2)=O)CN(C(=O)C2=CCCCC2)CCCO1 O=C(N=c1nc[nH]n2cccc12)N1CCCCC1CN1CCN(C2CC2)CC1 Cc1nn(C)cc1C(=O)N(C)CCOCCCNC(C12C=CC(CC1)C2)=O N1(C(C2(CC#C)CCOC2)=O)CCC(CF)(NC(=O)COCCCF)C1 C=CC(C(=O)N1CC(OCCSC)C1)NC(c1ccc(F)s1)=O c1(C(=O)NC2C(CO)CCN(C(c3c(C)nn(C)c3)=O)C2)cccc2cncn12 CC1(C)CCN(C(c2ccn(C(F)F)n2)=O)CC1NC(=O)CCOC1COC1 c1(C(N2CC(C=C)C(NC(C3COCCO3)=O)C2)=O)cc2sccc2n1C N1(C(C2(C(C)C)COC2)=O)CCCC(CCNC(=O)C(C2CCCCC2)F)C1 c1(C(=O)NCCC2CN(C(COC(CC)(C)C)=O)C2)nn(C(F)F)cc1Cl CCCCC1C(=O)NC2C(CC2)C(=O)N1.c1(C(=O)OCC)n[nH]c(C2CC2)n1 C(C)(CCCNC(C1CCOC1C(=O)O)=O)NC(CCC)=O c1(C(C(=O)NC(CC)C)N(CC(C)C)C)ncn(C)n1 N1(C(C2(Cl)C(C(C)=O)C2)=O)C2CCC(C2)C1C(=O)N(C)CCN(C)C(C)=O c1(C(=O)NC2CCN(C(C3=C(C)CCC3)=O)C(C)C2)coc2c(F)cccc12 C1(C)(C(=O)NC2CCN(C(COCC=C)=O)C2CC)CCC(F)(F)C1 c1(OC)ccc(O)cc1C(=O)NCC1CN(C(C2CCC2C(C)(C)C)=O)C1 C(CCF)(C(=O)NCC1COCC(C)O1)NC(CCC=CC)=O c1(C(=O)NCCC(C)NC(C2(C#N)CCCC2)=O)n[nH]c(Cl)c1Cl N1(C(c2nc(C(N)=O)sc2)=O)CC2(C1)CN(C(c1cc(C(F)(F)F)on1)=O)C2 C1(NC(c2ccc(CCC)[nH]2)=O)CC12CCN(C(=O)C1CC1)CC2 c1(C(N(C)CC2(CNC(C3CSCCS3)=O)CC2)=O)cc2c(nc1O)CCCC2 N1(C(C2C(C(=O)OC)C2)=O)CC2CC2(NC(c2oc(CO)nc2C)=O)C1 C1(CC)CN(C(=O)C(C)CN2CCCCC2)CCC1N=c1nc(C#N)[nH]cc1C C1(NC(CCC)=O)CC2(CCN(C(=O)C(c3ccccc3F)OC)CC2)C1 Cn1nc(Br)c2c(NC3CC(NC(=O)CN4CCCCCC4)C3)ncnc12 CC(C)C(F)C(=O)NC1CC12CC(NC(c1cccc(Br)c1)=O)C2 N1(c2snc(C(=O)OC)n2)CC2CCC1(CNC(C1CCCCO1)=O)CC2 C(C1=C(C(=O)OC)C(c2cccnc2)NC(=O)N1CCC#N)OC c1(NC(C2CN(C(c3cnc(Br)o3)=O)CCC2(F)F)=O)ccc2ccoc2c1 c1(C(N2CCC(NC(C(C)SCCCC)=O)C2)=O)ccc2c(C)noc2n1 N1(C(CCC)=O)CCCN(C(C2CC3(CCCN3C)C2)=O)C(C)C1 N1(C(c2c(C)sc(C)c2Br)C(=O)NC2COC2)CCC12CCN(C)C2 N1(C(CC2C(C)(C)CCO2)=O)CCC(C(=O)NC(CO)C2(C)CC2)C12CCC2 C1(C(=O)NC2(CO)CC(CO)C2)CCCN(C(C2CCOC2)=O)CC1 CCC(C(=O)N(CC(O)CN(C(=O)Cc1cn[nH]c1)C)C)Sc1nc(=N)[nH][nH]1 C1(NC(c2ccc(OC)c(F)c2)=O)CCN(c2ncc(C)cn2)CC1(C)C C1(C(=O)OC)CC(C(C)(C)C)CN(C(=O)CCCOc2cccc(Br)c2)C1 S(=O)(=O)(c1cc2c(cc1Cl)NC(=O)C2)N1C2CN(C(C3CC=C(C)CC3)=O)CC21 N1(CC(=O)NC2(C)CN(C(c3ccn(CC)c(=O)c3)=O)C2)C(=O)C(C)C(C)C1=O C#CCC(C)(C(=O)NC1CCCC(O)C1)NC(C1CCC(C)(C)OC1)=O c1(C(=O)NC2C(NC(Cc3cnn(C)n3)=O)CCCC2)c(F)cccc1[N+](=O)[O-] c1(C(=O)NC2CC3(C2)CC(CNC(C2CC24CC4)=O)C3)ccc2nnc(S)n2c1 C(c1cc(OCC)cc(OC)c1)=CC(=O)N(CCCN(C(CC(CC)C)=O)C)C O=C1CC(c2ccc3[nH]ncc3c2)=NN1CCC(F)(F)F N(C1CCc2cccc(F)c21)C(c1c[nH]c2c(F)cccc12)=O C1(NC(CN(C(C)C)C)=O)CC2CC1CN(C(=O)CC1(C)CCC1)C2 CC1CCC(C2OCCO2)N(C(=O)NCc2ccc(-c3ccncc3)cc2)C1 c1(C(N2C3C(C(N4CCC5(CCC5)C4)=O)C(C3)C2)=O)ccc(F)c(Br)c1F c1(SCC(=O)NCC(C2CCC2)NC(C2CCN(C)C2)=O)ccccc1F c1(OCC)cc(C(=O)N(C2CN(C(=O)COC(C)(C)C)C2)C)ccc1OC C1(CC)CN(C(=O)C2=CCCCO2)CCN1C(=O)C(C)Oc1cccc(F)c1 CCCCCCC(C)CC(=O)NC1(CNC(C2CCCCCC2(F)F)=O)CC1 c1(CNCC2(C)N(C(CSC(C)=O)=O)CCC2)cccc2c1CCCC2 C1(NC(CCCCC)=O)CC2CCC1N(C(c1nccc(C)c1O)=O)C2 N1(C(CC(CCC)C)=O)CCCCC2(CCN(CCS(C)=O)C2)C1 N1(C(CC=CCC)=O)CCCC(NC(=O)C(C)(C)C2CCC2)C1C N1(C(C(C)O)=O)CCCC2C1CCN2Cc1ccc(N2CCCCC2)cc1 C1(C(=O)NC(c2ccsc2)C)CCN1C1CCCC1 Cc1ccc(C(=O)N(C2CCCN(C(=O)C(C)Cc3cnc[nH]3)C2)C)c(N)c1Cl N#Cc1ccccc1N1CCN(C(=O)Nc2cc(-c3ccccc3)on2)CC1 Cn1cc(NC(c2ccnc(C(C)(C)C)c2)=O)cc1C(=O)NC(C1CCCC1)CO c1(C(N2C3CCN(C(CC=C)=O)CC3CC2)=O)cc(=NS(C)(=O)=O)cc[nH]1 C(=O)(CCCC(=O)N1CCC(CC(N2CCCCC2C2CC2)=O)C1(C)C)OCC N1(C(C2(CC)CCCC2)=O)CC2CS(=O)(=O)CC2(NC(=O)Cc2ccccc2)C1 c1(C(=O)NCC(CN(C(C(OC)OC)=O)C)O)cc(F)c(F)cc1C(F)(F)F c1(C(CC)C)ccccc1C(=O)NC(C)CNC(=O)C=CCN(C)C C1(C(=O)NCC2CCC(NC(c3c(C)scn3)=O)CC2)CC2CCCCC2C1 N1(C(c2cn(CC)nc2C)=O)CCC(NC(C2CCC23CCC3)=O)C(C)C1 Cc1ccc2cc(C(=O)NC3CCN(C(C4CC(O)C4)=O)CC3F)cn2c1 CCC(CC(=O)NCCN(C(=O)CC1CCC(C)(C)O1)CC)C(C)C C1(C(=O)Nc2ccccc2)CCCCCN1C(c1ccncc1C1CC1)=O C1(NC(c2c(C)nccn2)=O)CCN(C(=O)CCc2cc(F)ccc2F)CC1O C(=O)(CC(C)C(=O)N1CC(NC(c2ccccc2SC)=O)C(C)C1)OC c1(OC)cc(C)ccc1-c1ccc(NC(=O)NC(c2cccc(C)c2)=O)c(C)n1 Cc1cnc(C(C(=O)NC(C)(C)C)N(C(C)C(=O)OCCO)CC2(C)CC2)n1C Cc1nc(C)c(C(=O)NC2CC3(C2)CC3NC(=O)C=CI)o1 C1(N(C(C2CCN(C(C)=O)CC2)CO)C(=O)COCC(C)(C)C)CCS(=O)(=O)C1 c1(C(N2CCN(C(CCCCCC)=O)C(CCO)C2)=O)cc(Cl)c(F)cc1O c1(CC(=O)NC2CCCC(N(C(COCCC)=O)C)C2)cccc2sccc12 Cc1cnc(C(=O)NC(C)(C)CN(C)C(c2csc(C3CC3)n2)=O)cc1C c1(-n2ncc(NC(=O)NC3CC(OC)C3(C)C)c2C)ccc(Cl)cc1Cl c1(C(N2CCC(C)(CNC(C=CC=CCC)=O)C2)=O)cccc2nc(CC)sc12 N1(S(=O)(=O)c2cnn(CN3CCCC3)c2)CC2C3CCC(C3)C2C1 c1(C(=O)NCCOCCCNC(=O)CCC2CCOC2)ccc(OCF)cc1F c1(OC)ccc(OC)c(CNC(c2cccc(OCC#N)c2)=O)c1 Cc1nc2c([nH]1)CC(C(=O)NCC1(NC(c3ccc(OCF)nc3)=O)CC1)CC2 c1(OC)n[nH]c(C(C)NC(=O)NC2CCN(c3ccccc3Cl)C2=O)c1Cl Nc1ccc(C(=O)NC2(CNC(C3CCC(C(F)F)O3)=O)CCOC2)c(F)c1F c1(C(C)=O)cc(F)ncc1OCc1ccc(Br)cc1.c12cc(cn1C)NC(=O)N2 c1(C(N2CC3C(NC(CCN(C)CC)=O)C3C2)=O)cccc2c1CCC(=O)N2 c1(C(=O)NC2CN(C(CCSC)=O)CC3C2C3)c(C)ccc2c1CCCN2 C#Cc1cc(C(=O)NC(CN(C)C)CC(=O)NC2(C#C)CCCOC2)cc(F)c1 c1(C(=O)NCC(c2ccc(Cl)c(Cl)c2)C)ccc(F)cc1C1CC1 Cc1cc(F)ccc1C=CC(=O)NCC1CCCCN1C(=O)C(C)n1ccnn1 N1(C(COC(C)(C)C)=O)CCC2(CC(NC(=O)Cc3cccc(Cl)c3F)CO2)C1 CCC(CC)(CCOC)C(=O)NCC(C1CCC1)NC(C1CCC(CC)CC1)=O N1(C(C(C)NC(=O)NC)=O)CCCN(C(c2cc(C#N)on2)=O)CC1 CC1(C)CCC(CNC2CCN(Cc3ncccc3F)CC2)C1 Cc1nccc(NC(C)CC(C)NC(c2cnncc2O)=O)n1 c1(NC)ccc(C(N2CC(NC(=O)Cn3ccnn3)C(CC3CC3)C2)=O)c(Cl)c1 CCCCC(C(=O)NCC1(NC(=O)CN2Cc3ccccc3C2)CC1)C(C)C C(C(C)(CO)CC=C)NC(CC(CC)N(C(C1(C#C)CC1)=O)C)=O Cc1ccn2ncc(C(=O)NC3(CO)CN(C(=O)COCC(F)(F)F)C3)c2n1 Cc1n[nH]c(C)c1CCCNC(=O)CCN(CCO)C(C1NC(=O)OC1C)=O c1(CCNC(=O)NCCCOCOC)cnc2n1CCC2 c1(C(C(=O)NC)N(C)Cc2nc(CC)sc2)ccc(F)c(F)c1 C(C(C)(C(=O)SC)OC)OC.C=C(CNC(=O)N)CCNC(=O)OC(C)(C)C c1(C(=O)NCCCCCN(C(c2onc(C)c2C)=O)C)cnc2scnc2c1 C1(C(=O)OC(CNC(C2(CCNCCSCCOC)CC2)=O)(C)C)CCCC1O CCC(CC)C(C(=O)NCC(C)(O)CNC(=O)C(N1CCN(C)CC1)(C)C)OC c1(C(N(CCC(N2CC(=CCC)C2)=O)CCO)=O)n[nH]c2ccccc12 c1(C(=O)NC2C(NC(CCSCC(C)C)=O)C2)cnn2ccncc12 C1(CC)COC(C)(C)CN1C(=O)CC(CC(C)C)NC(=O)CC(C)n1cccn1 CC(C)(F)CCC(=O)NC1CC2(C1)CN(C(c1ccc(C(C)(C)C)s1)=O)C2 CCCCCCC(C)NC(C1C2CC2CN1C(c1ccn(CCC)n1)=O)=O N1(C(c2cccn3ccnc23)=O)CCN(C(=O)C2=CCCC2)C2CCCCC2C1 N1(C(C(CC)OC)=O)CC(NC(c2cn(Cc3cccs3)nn2)=O)C(O)C1 C1(C(C(=O)NC)N(CCOCCO)CC2CCOC2)CC12CCC2.CC c1(C(=O)NCC2CC(NC(c3ccc(C(C)=O)s3)=O)C2)ccc(Cl)nc1 C1(CNCC(CC)(C)c2ccncc2)CCC2(CCC2)CN1C N1(C(C(F)OC)=O)CC(NC(=O)CSC(C)C)C(C)(C)C1 N1(C(C(C)NC(=O)C(C)(C)C)=O)CCC2C1CCCN2C(=O)C(F)=C1CCCC1 C1(CNC(c2nc(CCC)oc2)=O)CN(C(c2ccc(C)nc2N)=O)CCN1C n1(CC)ncc(C(=O)NC(C)(C)CN(C)C(c2csc(-c3ncc[nH]3)n2)=O)n1 C1(NC(CC(c2ccc(OC)cc2)(C)C)=O)CCC2CN(C(C)=O)CCC2C1 C(CCCCCCC(=O)NCCCN(C)C(C1COC(=O)N1C)=O)SC N(C1COCc2cc(OCCNC)ccc21)C(=O)Nc1n(C(CCC)C)ncc1 Cc1oc(CNC(=O)CCn2ccnn2)nc1C(=O)NCC1CSC1 c1(C(=O)NC2CN(C(C=CC(=O)OCC)=O)C(C)CC2)nc2c(s1)CN(C)CC2 CN1CCC(NC(=O)C(c2ccc(Cl)cc2)(C)C)C1(C)C C1(NC(C2=NOC(C)C2)=O)CN(C(C2CCC(=O)CC2(C)C)=O)C2CCCC12 N(C(=NCC(C)C)N(C)Cc1nc2cc(F)ccc2o1)CC1(OC)CC1 C(=O)(C(O)CCC(C)C)NCC1N(C(Cc2cc(C)no2)=O)CC=C1 C1(O)(CC)CCN(C(=O)C(c2cn(C)nn2)NC(C2CC2CC(C)C)=O)C1 C12CN(C(=O)C=CCOO)CC1C2.c1(NC(C(C)C#N)=O)ccc(F)cc1 C1(NC(c2ncsc2Br)=O)(CNC(C2(O)CC2)=O)CCOC1 CC(O)C(C)(C)C(=O)NC(C)CCN(C)C(c1cc(F)n(C)n1)=O c1(C(=O)NC(CCC)Cc2ccccc2)coc2c1N(C)C(=O)CCC2 Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(C23CC(CC(C)O2)C3)=O)cc(C)n1 C1(NC(CC2CN(C)C2)=O)CCC12CCN(C(C1(C)CCNC(=O)C1)=O)CC2 C1(NC(COCc2cc(C)on2)=O)CN(C(=O)C(O)CN2CCC2)CC1N=[N+]=[N-] c1(C(N2C(CNC(C3CC4C=CC3C4)=O)CC2)=O)ccc2c(c1)CCCS2 c1(OC)c(C(=O)NC2CN(C(=O)C(c3ccccc3)O)CC2(C)C)cccc1Cl N1(C(CC2N(CC)CCC2)=O)CCOC(C(C)NC(=O)CNC(=O)OC)C1 N1(C(c2c(C)cn(C)n2)=O)CC(NC(C2(Br)CC2)=O)CC12CCCOC2 C1(c2ccc(OC(F)F)cc2)CN(C(=NCC=C2CCC2)NCCOC)CCS1 Cc1ccnnc1C(=O)NC(C1CCCC(CC(N2CCC2(C)CCO)=O)C1)O c1(NC(C2(OC)C(CC)CCCC2)=O)cccc(S(C)(=O)=O)c1C C1(CNC(C(CCC)OC)=O)CN(C(c2cc(C(F)(F)F)n(C)n2)=O)CCN1C C1(NC(N2CCN(c3ccc(Cl)cc3)CC2)=O)(CO)CC2C=CC1C2 c1(C(N2C(COC)(CNC(=O)C(F)F)CCC2)=O)cc2c(N(C)C)cccc2s1 c1(C(C)C(N2CCC(N(C(=O)Cc3cnns3)C)C2)=O)c(F)cccc1F C1(C(C)NC(C=C(C)C2CC2)=O)CCCN(C(c2ccc(Cl)o2)=O)C1 c1(C(=O)OC)nc2cc(-c3c(C)ccc(C#C)c3)c(OC)cc2n(C)c1=O c1(CCC)ccc(N2CC(C(=O)Nc3ccnc(C4CC4)c3)CC2=O)cc1 C1(C(N(CC(C)CNC(=O)CC2CCNC(=O)C2)C)=O)CCC(C)(C)CC1 C1(C(C(=O)NC2C(C(C)C)CCC2)C)CCN(C(=O)COC2CC=CC2)CC1 c1(C(=O)NCC(C)N(C(c2ccc(F)cc2F)=O)CC)cccn2cnnc12 C1(CNC(C=Cc2scc(C)n2)=O)CC(C)(C)CN1C(C1CCOC(CF)C1)=O c1(C(=O)NCC(CC)NC(C(CC)c2ccccc2)=O)n[nH]c2c1CCOC2 c1(-c2ccc(-c3n(CCC4C(C)C4)ccn3)cc2)ccc(Cl)c(C(F)(F)F)c1N N1(C(C(CC)=O)=O)CC2(CCN(C(=O)C(C)=C3CCC3)CC2)C1 CN=c1[nH]c(=NCc2cccc3c2OCC3)[nH]c(=NCc2cc(F)cc(F)c2)[nH]1 N1(S(CC#N)(=O)=O)CCC(c2ccccc2)C(O)C1.c1(N2CC2)ccc(I)c(Cl)c1 c1(C(N2C(C(=O)NCc3c[nH]nc3-c3ccccc3)CC2)=O)cccc(F)c1F c1(CC)cc(C(=O)NCC(C)CN(C)C(C2CSCCS2)=O)ccc1Cl c1(C(C=C=C)C)nc(C2CCOC2)nn1-c1ccc(CC)cc1 c1(C(=O)NCC2CCCCC2NC(C2COCCO2)=O)cc2n(n1)CCCC2O C(=O)(CC(C)CC(C)(C)C)N1CC(NC(Cc2cc(C)on2)=O)C(C)(C)C1 C1(NC(=O)NOCCC(O)COC)CCC(C(=O)N(C)C)CC1 c1(COCC(C)(CO)NC(C)CCCOc2ccccc2)ccc(Cl)cc1 CN1C(=O)CC(C(=O)N(CC)CC2CC2NC(=O)Cc2ccc(Cl)nc2)NC1=O c1(NC(N(C)CCOc2ccccc2)=O)ccc(C(C)(C)C)cc1Br c1(C(=O)NCC(CC)NC(CCCC#CC)=O)cc2ccccc2cc1O N1(C(c2ccccc2)C)C(=O)NC(c2cnn3c2CCC3)C(C(=O)OC)=C1CCl N1(C(c2c(CC)csc2)=O)CCOC(C(C)NC(=O)CNc2cccnc2Cl)C1 C(C)(C)(CCCC(=O)NCC1CC1[N+](=O)[O-])NC(C1(COC)CCCO1)=O C1(C(N(CC(C)NC(=O)C(=O)NC2CC2)CC)=O)(CSC)CC=CC1 C1(NC(c2ccc(NC(C)=O)cn2)=O)CN2CCCN1CC2 n1(CC)ccc(C(=O)NCCC(C)N(C)C(c2cc(C)c[nH]2)=O)cc1=O c1(CC(=O)NC2C(CNC(=O)CSC(F)(F)F)C2)c(F)cccc1Cl C1(C(N)=O)(NC(Cn2cc(Cc3ccncn3)nn2)=O)CCOCC1 c1(NC2CC(NC(N(C)CC)=O)C2(C)C)c(C)ccn(C)c1=O C(=O)(C1=CCCOCC1)N1CCC(O)(C(C)NC(=O)CCS(=O)(=O)N(C)C)C1 Cc1nonc1CC(=O)N(CC(=O)NC(Cc1ccco1)CO)C C1(NC(=O)NC2C(COC)(CO)CC2)CCC(P(C)(C)=O)C1 c1(NCC2N(C(C3C(c4cn(C)nn4)C3)=O)CCC2)nc[nH]c2nccc1-2 C(CNC(=O)C=CC1CCCCCC1)(CC(F)(F)F)NC(c1n(C)cnc1)=O n1(CC)cc2cccc(NC(=O)NCC3CNC(=O)CO3)c2n1.NC CC(C(C)C(=O)N1CC2CCC1CN2C(=O)C=CBr)S(C)(=O)=O N1(C(C(C2CN(C(=O)C(O)C(C)C)C2)C2C(C)C2)=O)CCC(C)C(CO)C1 c1(C(=O)NCC2CCC(NC(C3C(C)=C3)=O)C2)n[nH]c2cc(C)ccc12 CC1CC(NC(c2c(Cl)n[nH]c2C2CC2)=O)CN(C(=O)CC2CCOCC2)C1 c1(C(=O)NCCCCc2cn(-c3n(C)nnc3)nn2)ccc(C2CC2)cc1 C1(N(C(=O)CCCc2ncco2)CC(=O)NCCF)CCC(=O)NC1=O Cc1ccc(C(N2CCC(CC(=O)Nc3ncc(Cl)nc3Br)C2)=O)cc1Br N1(C(c2cc(OC)n[nH]2)=O)CCCCC12CC(NC(c1cc(CO)on1)=O)C2 N1(C(c2[nH]ccc(=N)n2)=O)CCC2(NC(=O)Cc3ccc(Br)nc3)CCCC12 C1(O)(CNC(C(c2cnn(C)c2)C)=O)CCN(C(c2cccnc2S)=O)CC1 c1(C2(O)CC(NC(c3cnc(OCC4CC4)s3)=O)C2)ccc(Cl)cc1 C(=O)(C(CCC(C)C)NC(c1sccc1CO)=O)NCc1nnc(C)o1 N1(C(COCC)=O)CCC2(CCC(NC(c3c(SC)cnn3C)=O)C2)CC1 c1(C(N2CCCCC(N(C(=O)C(N)=O)C)C2)=O)c[nH]c2cccnc12 N1(C(CC2CCCC(OC)C2)=O)CCC(C)(O)CC1.c12cc(on1)C(=O)NC2 CS(=O)(=O)C1CCC(NC(C2CC(=O)N(c3cccc(Cl)c3)C2)=O)C1 Cc1cncc(CC(=O)NC2CC(C)(NC(c3csc(-c4nc[nH]n4)n3)=O)C2)c1 N1(C(C2CC(OCC)C2)=O)CC2(C1)SCCC2NC(C1CC1C(C)(F)F)=O C1(F)(CNC(c2csc(C(F)(F)F)n2)=O)CCCN(C(C2CCOCC2)=O)C1 c1(C(CNC(CC)(C)C)C2CC2)ccc(C)cc1C1CC1 O=C(CC1NC(=O)c2ccccc21)NCCN(C(c1ccon1)=O)C1CC1 C1(NC(=O)C=Cc2ccc(O)cc2)CC12CCN(C(c1n[nH]cc1F)=O)CC2 n1(CC(=O)N(C)CC2(NC(c3c(CCC)[nH]cc3)=O)CC2)ncc(O)nc1=O c1(C(=O)NC(C2CN(C(C3C(F)(C(=O)OC)C3)=O)C2)C)cc2n(n1)CCCO2 c1(C(N(CCNC(C23CC(C2)C(C)O3)=O)CC)=O)cc(C)nc(C)n1 c1(C(C(F)(F)F)OC(c2cccc(CC3CC3)n2)=O)ccc(F)c(Cl)c1 N1(C(C2(F)CCCC2)=O)CCN(C(C2CC2C(F)(F)F)=O)C(c2ccccn2)C1 N12CCCC(CO)(C1)NC2=O.c1(Nc2nccc(C(F)F)n2)cc(Cl)nc(Cl)c1 c1(C(N(CCCNC(C(CC2CC2)OC)=O)C2CC2)=O)cc(C)cc(F)c1 Cc1cnn(C)c1C(=O)NCC(C)CC(=O)N1CC2C(C(N)=O)C2C1 C1(NC(=O)NCCC2(C(=O)NC(CC)C)CCCC2)C(C)(C)C1(C)C N1(C(C=Cc2cc(C)no2)=O)CCC2CN(C(=O)C(O)CC(C)C)CC2C1 N1(C(CC(C(C(C)C)C)C)=O)CCc2ccccc2C1CNC(c1cc[nH]n1)=O c1(C(C(=O)NCCCSC)N(CCCC(C)C)C)cc(-c2cccnc2)nn1C CN=S(C)(=O)c1cccc(C(N2CCCCC2CNC(c2coc(Br)n2)=O)=O)c1 C1(NC(C(C)C(c2n[nH]cc2Br)c2nnnn2C(C)(C)C)=O)CCCSCC1 C1(NC(C=CC=CCC)=O)CCN(C(=O)C(C)(C)c2cnco2)CCC1CO c1(C(N2C(CN(C)C(c3ncoc3Br)=O)CCCC2)=O)ccc(F)cc1F C1(NC(c2ccc3cc(OC)[nH]c3c2)=O)CCCCC12CCCN(C(C)=O)C2 C(=O)(CC(O)CC(C)(C)C)NCC12N(C(C(C)NC(CC)=O)=O)C(CC1)CC2 C12CC3(C1)CC3C(=O)NOC(C1CC1)C(=O)N2.C1(N)C(C#N)C1(C)C.CCO c1(C(N(CC(CN(C(CCC#C)=O)C)O)C)=O)cc(N)ccc1Cl C(=O)(C(C(C)(C)C)NC(C)=O)N(C)CC1N(C(CNC(C)=O)=O)CC(F)C1 N1(C(C(C)OCCCC)=O)CCN(C(=O)C(CO)C(C)C)C(C2CC2)C1 C(=O)(C(F)CCC(C)C)NC1(C(=O)NCC(COC)C(C)C)CCCC1C CC(CNC(C1CCC1(F)F)=O)(Cn1cccn1)NC(=O)CSC(F)F C(C(=O)NC1(OC(C)C)CCC1)(C(C)C)NC(COCC(=O)NC)=O N1(C(c2nc(C)sc2)=O)CC2CCCN(C(=O)Cc3csc(NC=O)n3)C2C1 N1(C(C(COCC)C)=O)CCOCC1(C(=O)N(C)CC1COC(=O)N1)CC CN1C(=O)CSC1=CC(=O)NCC1CCN(C(=O)CCC2CCCC(=O)N2)C1 C1(CCC)(NC(=O)C(C)C(O)CC)CCCN(C(c2c(Cl)cnn2C)=O)C1 c1(NC(C(=O)NCC2CCSC2)=O)cc(C(F)(F)F)cc(Cl)c1 C(CC(C(C)C)NC(=O)C(c1cccc(F)c1)F)N(C(C1C(CC)C1)=O)C N1(c2cc(C(C)C)ncn2)CC2CC1CN2C(=O)COc1ccc(Cl)cc1 c1(C(=O)NCCC2CC(NC(CC(CC=C)(C)C)=O)C2)ccc2oc(C)nc2c1 N1(CCN(CCNC(CC(=O)OC)=O)C(c2ccncc2)=O)CCN(C)CC1 CCC(CC)C(F)C(=O)N1CC(C(N2CCC(NC(=O)NC)C2)=O)CC(C)C1 C1(CN(C(=O)CCCN(C)C(C2CCCO2)=O)C)CCCOC1 N1(C(c2c(C)noc2C)=O)CCC2C(NC(c3ccc(-c4ccco4)s3)=O)C1C2 C1(C)(OCc2cn(CCC=C)nn2)CCCN(C(C2(C)CCNC(=O)C2)=O)C1 c1(C(N2CCC(CN(C(=O)C=CC3CC3)C)C2)=O)cc(F)cc2ccncc12 c1(C(N2C(C)C(NC(=O)Cc3csnn3)CC2)=O)cc2cccnc2s1 C1(CNC(c2c(C)oc(Cl)n2)=O)CN(C(=O)COC2(C)CCC2)C2CCCCC12 c1(C(=O)NCC(CC=C)NC(C2CCN(C3COC3)C2)=O)cc(C)cc(O)n1 C12(CNC(c3ccc(C(F)F)cc3)=O)CC1CN(C(C1C(F)(F)C13CC3)=O)C2 C1(C(=O)NCC(c2cccs2)O)CCN(C(C2(C3CCCO3)CC2)=O)C1 C#CC1(C(=O)N(CCCCCC)C)CCN(C(c2ccc(OC)s2)=O)C1 C(=O)(C(CNC(c1cnnc(O)c1)=O)C(C)(C)C)NCCCc1cnc(C)o1 Cc1cc(C)c(CNC(=O)CC2(C)CCN2C(C2CCCC(=O)CC2)=O)cn1 C=CCC(C)(C)C(=O)NC(CNC(c1ncsc1C)=O)C(C)C(C)C C1(CNC(c2ccc(C3CC3)s2)=O)CCN(C(=O)CC2CCSCC2)CC1(F)F c1(C(=O)NC2CC(CNC(C3(CC)CCNC3=O)=O)C2)ccc2c(C)noc2c1 C(C)(C(CC(=O)NCC1CC1C(C)C)NC(C1C(C)C1C)=O)OC CC(C)(CC(=O)N1CCOCC(NC(=O)CC2CC(=O)NC2=O)C1)C(F)F CCC1=C(C(=O)N2CC(CNC(c3[nH]nc(C(F)(F)F)c3C)=O)CC2C)SCCO1 c1(CC(N2C(CCCNC(C(CC)F)=O)CCC2)=O)ccc2nonc2c1 c1(C(=O)NCCC2CCN(C(C(F)=CC)=O)C2)cc2cc(F)cc(F)c2nc1C CCC1=C(C(=O)N2CCCC(CN(C(=O)C(O)C(C)C)C)C2)SCCO1 O=S(=O)(C(F)F)C1CN(S(=O)(=O)c2ccccc2CF)C1 C(=O)(C(F)(F)C(C)O)NCC1C(NC(c2c(COC)cco2)=O)C1 c1(SCCNC(=O)NCC(CF)SC(C)C)ccccc1 c1(CC(=O)N(CCN(C(C(C)OCCCC)=O)CC)CC)cc(C(C)C)nn1C c1(CCC(=O)NC2(COC)CCN(C(CSCCC)=O)C2)cnc2ncccn12 CC1(C)OCCC1NC(c1ccc(CNC(C2(C#N)CCCO2)=O)s1)=O n1(CC(C)C)cc(C(=O)NC(C)(CNC(C23CCC2C3)=O)C2CC2)cn1 c1(NC(c2nc(C)[nH]n2)CO)cc(CO)nc(CNCC2(N3CCOCC3)CC2)n1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CCN(C(=O)C=CC3CCCO3)CC(C2)C1 O(NC(=O)C(C)C(C)NC(c1ncn2ccccc12)=O)CCOCC#C c1(OC)ccc(C(=O)NC2CCN(C(c3cc(C)n(C(F)F)n3)=O)CC2)nc1 C(=O)(C(C)(F)CC1CCCC1)NCCCN(C(c1c(C)scn1)=O)C1CC1 C(=O)(C(F)C(C)(F)F)N1CC(C)(NC(COCCC)=O)C1 N1(CC)CCN(CC(=O)NC(C(=O)N2CC(n3ccnc3C)C2)C2CCC2)CC1 c12cnc3c(cnn3C(=O)N1CC)c2.C1(CO)CCN(C(c2ccsc2)=O)CC1 C=CCC(C)(C)CC(=O)NC1CC(O)C1CC(N1CC2(CCC(=O)O2)C1)=O C(=O)(C1=CCCN(C(=O)OC(C)(C)C)C1)N(C1CCCC(O)CC1)C c1(C(=O)NCc2c(C(N3CC(NC(CC)=O)C3)=O)c[nH]n2)cc(C)n(C)c1 C(=O)(C#CC1(C)CCCO1)N1CCCC(N(C(c2cn(CC)nc2)=O)C)CC1 C1(C(=O)OC)CCCCC1C(N1CCC(N2CCCC2)C1)=O.c12scnc1N2 c1(OCC)cccc(NC(c2nc(C(=O)Nc3ccc(C)cc3)cs2)=O)c1Cl C(=O)(CC(CC)CCCC)N1C(C(=O)NCC#C)C2CC2C1.c12ccnc(c1)C2 N1(C(c2occ(C)c2C)=O)CC(C2CCCN(C(c3csc(Cl)n3)=O)C2)C1 N1(C(CN2C(C)CCC2)=O)CCCC(CCCCNC(C23CC(C)(CO2)C3)=O)C1 c1(OC)cc(Cl)ccc1C(=O)C(=O)NCCC(C)NC(c1ccc[n+]([O-])c1)=O c1(CC(=O)NCC2OCCN(C(C3CN(C)C(=O)N3)=O)C2)cn2c(n1)CCCC2 CCCC(CNC(C1(NC(=O)CC(C)(C)OC)CC(F)(F)C1)=O)CCO C(N=c1cc(C)nc(N2CCC(C3CCCO3)CC2)[nH]1)C1C(COC)C1 C(=O)(C1=NOC2COCC12)NC1(CC)CN(C(c2csc(-c3ccoc3)n2)=O)C1 C(=O)(C(C)CN(C)CCC)NCC1C(CC(=O)NC(CCC)C2CCC2)C1 c1(NCc2n(C(C)C)ncn2)[nH]c(=NC2CCCC2N(C)C)nc2ncn(C)c12 n1(CC)c(C)c(C(N2CC(OC)CC(O)C2)=O)c2cc(OC)ccc12 c1(C(=O)NCC2(O)CC(NC(CCC=C(C)C)=O)C2)ccc(Br)c(C)n1 C1(CC(=O)N(C2CCN(C(c3ccc(C)nc3)=O)CC2)CC)CCC(C)CO1 c1(OC)ccc(F)cc1NC(C1CC1NC(c1nc(C)no1)=O)=O N1(C(CCCCCC)=O)CCC2CN(C(=O)CC3CCCOC3)C2C1 N1(C(CCN(C(C)=O)C)=O)CCC(OCCNC(C2CC=C(C)CC2)=O)CC1 C(CN=c1[nH]c(C(=O)N(CC(F)(F)F)CCO)cs1)c1c(Cl)c(C)n(C)n1 C1(N(C(CC=C)=O)CC2CC2)CCN(C(c2ccccc2OCC=C)=O)CC1C C(=O)(CC1OCc2ccccc21)N1CCN(C(c2c(C#N)nc[nH]2)=O)CC(O)C1 Cc1nn(C)cc1CC(N1CC(CNC(C23CC(CN2C2CC2)C3)=O)C(C)C1)=O O=C(CCC(CF)CF)NCC1(NC(C2CCOC2C2CC2)=O)CC1 Cc1[nH]c2ccccc2c1C(=O)NC1CC(NC(=O)C=CC(C)C)C12CCC2 C(C(CO)(CO)NC(=O)CC1CCCOC1)N(C)C(c1cc(CO)on1)=O C1(O)(CNC(=O)CSc2cccc(F)c2)CCN(C(=O)C(O)CC2CC2)CC1 C1(C(=O)NCCC=CCCC)CN(C(=O)CC2CC(F)(F)C2)CC1(C)C c1(C(=O)NC2(CNC(c3ccc(OC)cc3)=O)CC2)oc2c(C)cccc2c1C c1(NC(C)CN2CCCC2=O)[nH]c(=NCCC2CCSC2)nc2scnc12 N1(C(c2scc(C(C)=O)c2)=O)CC(C)OC2(CCN(C(C3CC3F)=O)CC2)C1 C(=O)(C1CCCc2ncnn21)N1CCCC(CNC(CS(=O)(=O)NCC)=O)C1 N1(C(C23CCC(C)(C2)CO3)=O)CC2(COC(CNC(=O)Cc3cccs3)C2)C1 C1(C(N(CC(=O)Nc2cnn(C)c(=O)c2)CCC)=O)CC(=O)N(OC)C1 c1(OC)ccccc1SCC(N1CC(NC(c2cccs2)=O)CC1C)=O O=C(Nn1nnc2c1CCCC2)C1CCc2c[nH]nc2CN1C(C1CCSC1)=O N1(C(C=CC(CC)C)=O)CCCC(N(C(=O)CS(=O)(=O)N(CC)CC)CC)CC1 CCCC(C)(O)CC(=O)NC1(C)CC(NC(C2CC(=O)N(CC)C2)=O)C1 N1(C(C=CC(=O)OCC)=O)CCC2(CC1)CN(C(C)CNC(C)=O)C2 c12c(ncnc1Cl)N1CCC(C1)CNC2=O.C(=O)(C(C)S(N)(=O)=O)OC c1(C(=O)NC(C)CN(C)C(C2CC2C(F)F)=O)cc2cc([N+](=O)[O-])ccc2[nH]1 c1(C(=O)NCC(C)NC(C(C)NS(CCCC)(=O)=O)=O)nc2ccccc2s1 Cc1cc(C(=O)NC2CC(C)(CNC(C3CCCCC3(F)F)=O)C2)nc(O)n1 N1(C(C2CC3CC3N2C(=O)CC2CC(CF)C2)=O)C2CCC1CC1(CC1)C2 Cc1cc(C(C)CNC(N2CC(=CC#N)C2)=O)cc(F)c1 N1(C(C(=O)NCCSC)C2C(CC)C2)CCC(O)(CSC)CC1 c1(C(=O)NC(CNC(c2n(CC)ccc2)=O)C2CCC2)coc(C#N)c1 N1(CC)CCOCC1C(=O)Nc1cn[nH]c1.c1(N(CC)CC)ncc(C(C)=O)cn1 C1(C(N)=O)CCCC(NC(c2sccc2CNC(c2cccn2C2CC2)=O)=O)C1 n1(CC)cc(CC(=O)NCC2(C(=O)NC3CC3(c3ccccc3)C)CCC2)cn1 C1(C(=O)NCCCNC(C2(CSC)CCC2)=O)CSc2ccccc2O1 C(=O)(CCC(C)NC(c1ccn(C)n1)=O)NCCCOC(=O)NC CC1C(O)CCCN1C(=O)COC1(C)CN(C(=O)C(O)CO)C1 C(C#CC(=O)N1CCCc2nccn21)NC(C(C)(C)C#N)=O c1(N2CCC3(CCCN(C)C3)CC2)nc(=NC2CCOC2)[nH]c2c1SCC2 C(=O)(C1=CCN(C(C2(n3cnnn3)CC2)=O)C1)N1CC2CC(C(N)=O)(C1)C2 C1(C(N(C(C)CCNC(=O)CC2CC3(CC3)C2)C)=O)CCOC1(C)C C1(NC(C(CCSC)NC(N)=O)=O)CN(C(c2cnoc2C)=O)CCC1F N1(C(CNC(C2(N(C(C(C)n3ccnc3)=O)C)CC2)=O)C)CCOCC1 C1(CNC(c2ccc(Cl)s2)=O)(CNC(=O)C(C2CCCCC2)O)CC12CCC2 c1(C(c2nnnn2C2CCOC2)NCC2C(C(=O)OC)CC2)cc(C)ccc1Cl C(=O)(C(CCSC)NC(C1COCCO1)=O)NCC(C1CCC1)OC Cc1ccc(NC(=O)CN(C)Cc2ccccc2CN2CCN(C)CC2)cc1 Cc1cc(F)ccc1C(N1CCCCC(NC(=O)COCc2nc[nH]n2)C1)=O c1(C(=O)NC(CCOC)CNC(C2CC23CC3)=O)ccc(C)c([N+](=O)[O-])c1 CN1CCOC(C(=O)NC2CN(C(=O)CCc3cnc[nH]3)CC2O)C1=O C1(C(=O)NC(C)CCNC(c2ccncc2O)=O)CC2CCCCCC12 C1(C(=O)NC2(CC(=O)NCc3ccc(N(C)C)nc3)CCC2)CC2CC(=O)C1O2 C(=O)(C(CC)CC(F)F)N1CC(CC=C)(C(=O)NCc2cc(=N)[nH]cc2Br)C1 c1(CC(=O)NC2C(NC(c3ncc(C)nc3)=O)CCC2)cn2c(n1)CCCC2 C1(C(=O)NCC2(COC)CN(C(=O)CC3CCCO3)C2)CC2CC(O)CC(C1)C2 N(C1CCSc2ccc(F)cc21)C(C(=O)N(C(C)C)C)=O.C(CCN(C)CCN)N N1(C(c2ccnc(CC(C)C)n2)=O)CCN(C)C(CNC(c2cscc2Cl)=O)C1 N1(CC(=O)NCCC(=O)NCC2CC2)CCC(F)CC1.C12(CC1)C(=O)NC2 C=C(C)C(CC(=O)N1CC(NC(=O)CCc2ccc[nH]2)C2(CC2)C1)OCC c1(OC)cccc(OC)c1CC(c1ccc(C)nc1C)c1nnnn1C1CC1.NC c1(CN(C(CC)CN)Cc2ccccc2)ccc(C(C)(C)C)cc1 C1(C(N2CC(C(C)NC(c3cnsn3)=O)C2)=O)CC2(CC2)CN1C C#CC1CN(C(=O)Cc2nc(C)sc2C)CCN1C(c1cc([N+](=O)[O-])c(C)s1)=O c1(OC)cc(-c2cn(CC3CCCN3C(C3SCCCS3)=O)nn2)ccc1F Cc1ccc2c(c1)CCC(C(=O)NCCSCC1CCC(C)O1)O2 N1(C(CNC(CC)=O)=O)C2CCC1CC(CC(=O)NCC(C)(C)SC)C2 c1(C(=O)NC2C3N(C(c4ccn(CC#N)n4)=O)C(CC3)C2)ccc2c(c1)CCC2 c1(CCN(C2CCN(c3cc(C)ncn3)CC2)C)ccc(Cl)cc1F c1(C(=O)NCC2(O)CN(C(c3n(CC)ncc3)=O)C2)ncccc1Cl CCCCC(C(=O)NC(C)COCC)NC(=O)Cc1cccn1C N1(C(C(CC)N(C)C)=O)CCCC(NC(c2ccc(OC(F)F)cn2)=O)C1 N1(C(c2ccc(C=C)o2)=O)CC2OCCN(C(C3(C)CCCCCCC3)=O)C2C1 c1(OC(CNC2CN(C(COC(CC)C)=O)C2)C)ccccn1 N1(C(C2(OC)CCC2)=O)CC=CC(NC(=O)CCCn2cccn2)C1 C(=O)(C(C)(C)CC(F)F)NC1CCN(C(CC(COC)(C)C)=O)C(C)C1 C1(CC(C)(C)C)CN(C(C2CCC3(CC3)C2)=O)CCN1C(c1csc(C#N)c1)=O CC1C(NC(c2cccc(=O)o2)=O)CCCN1C(c1cc(C(F)(F)F)ccn1)=O Cc1ccc(O)c(CC(=O)NCCOC2CN(C(=O)C(C)(C)CC3CC3)C2)c1 C1(NC(=O)C(=O)NC2CCCO2)CCN(Cc2ccccc2CO)CC1 N#CC1(c2nnnn2C)CCC(C(F)(F)F)(NC(CCc2ccc(O)cc2)C2CC2)C1 N1(C(CCCCC)=O)CCC(NC(c2ccc(OC)cn2)=O)C(CO)CC1 C(=O)(C1COc2ccccc21)NCC1(O)CCCN(C(c2c(CC)nco2)=O)C1 C1(CC(=O)NC2(C)CC(NC(=O)CSCc3ccccn3)C2)CCCNC1=O c1(C(C)CCn2cc(CC(C(=O)O)NC(C3(C)CC3)=O)nn2)nncn1C N1(C(C(COC)N(C)C)=O)CCN(C(c2cc(O)n(C)n2)=O)C(CC(C)(C)C)C1 C1(NC(C2(N(C(CNC(C3C(C)C3)=O)=O)C)CC2)=O)CCCCC1(C)O C=CCCCC(C(=O)NC(C)(C)CC=C)NC(c1nccnc1N)=O C12(NC(=O)CC3CCC(O)C3)CCCC1N(C(C1CC3(CC3)C1)=O)CCC2 c1(OCC(=O)NC2CCN(C(C(CC)C#N)=O)C2)ccc(F)cc1O C(=O)(C(O)CC(F)F)N1CC(NC(CC2CC(=O)NC2=O)=O)(CO)C1 N1(C(c2ccc(SC)s2)=O)CCC(NC(C2CCN(C)C2=O)=O)C(CO)C1 Cc1cc2cc(C(N3CC4CCN(C(c5ccsn5)=O)CC34)=O)c(Cl)cc2[nH]1 c1(C(N2CC=CC(NC(c3n(C=C)nnc3)=O)C2)=O)cnn(C)c1S(N)(=O)=O c1(C(=O)NCC2(CN(C(CCCOC)=O)C)CC2)cc(F)c(C(F)F)cc1F C(=O)(C1=CCCCC1C)NC1(CC=C)CCN(C(=O)CCCC(F)(F)F)C1 N1(C(C2C(CC(C)C)C2)=O)CC2CC2(CNC(c2cn(C)nc2C(C)C)=O)C1 c1(OCC(=O)Nc2ncc(C)s2)ccc(-c2ccoc2C)c(F)c1 Cc1noc(Cl)c1CC(N1CCC(C)(CNC(C2(C)CC(C)(C)C2)=O)C1)=O CN1CC=C(CC(=O)NCC2(NC(c3cccc4c3C(=O)NC4)=O)CCC2)CC1 C1(NC(c2nc(C)c(C)s2)=O)CN(C(C2CCC(C)C2)=O)CCC1C C(=O)(CCC(CF)CF)N1CCC(CNC(C(NOC)=O)=O)C1(C)C C1(NC(C(F)=C(C)C)=O)CC2CCC(C1)N2C(c1ncc(C(F)(F)F)cc1N)=O C1(C(=O)NCC23CC(NC(=O)CC45CCCC4C5)(C2)C3)CCS(=O)(=O)CC1 CC(O)CCCC(=O)NCC1CN(C(=O)CSCc2cccnc2)CCO1 c1(OC(CC)C(=O)NC23CC(C2)N(C(=O)CCF)C3)ccc(C#N)cc1 C1(N(C(CC2(C=C)CCC2)=O)C)CCCN(C(=O)CC2CCC(C(F)(F)F)O2)C1 C=C(C)CC(=O)NC(C)(CNC(=O)C(C)COc1ccccc1)CC N1(C2C3CN(C(CC(C)NC4CC4)=O)C(C3)C2)CC(=O)NC2(CCCC2)C1 CN1CCCC(C(C)(C)NC(=O)NCC(C(F)(F)F)N2CCOCC2)C1 C1(C(N(C(CCCC)C)C)=O)C=CCN(C(C2(O)CC2)=O)C1 C(C(=O)NC(=O)NC(C)(C)C)N(C(=O)CC1CC1)C(C)C.OCO C(=O)(C1=NN(C)C(=O)CC1)N1CCC2(C(NC(CCC(C)=O)=O)C2)CC1 C1(C)(CNC(Cc2ccc(C)cc2)=O)CN(C(=O)C=C2CCC2)CC1C Cc1cc(C(=O)NCC2CCN(C(c3c(C)[nH]c(C)c3C)=O)C2)ccc1Cl c1(-n2cco2)nnc(N2CCC(NC(c3ccsc3)=O)CC2)n1CCN1CCCC1 C(=O)(C1CCc2c(Cl)cccc21)N1CCC(C(CNC(C2(CC)CC2)=O)F)CC1 CC1(C)CN(C(=O)C=CC(F)(F)F)CC1C(N1CCC(C)(O)C1)=O Cc1c(NCC(=O)N(CCCN2CCCC2=O)C(C2CCCCC2)=O)cnn1CC C(=O)(C1Cc2ccccc21)NC(C1(O)CN(C(c2c(N)ncc(C)c2)=O)C1)C c1(CCNC(c2n(C(CC)C)nnn2)c2ccsn2)ccc2c(c1)CCCC2 c1(CC)cccc(NC(=O)NC(C)CC2CCN(C)CC2)c1C c1(C(=O)N(C(C)(C)C2CC2)C)cccc(OC)c1O.C1(OC)CC(C(=O)NCCOC)C1 c1(C(N2CC(F)(CNC(c3c(C)nc(C(C)C)s3)=O)C2)=O)cccc(S(C)=O)c1 CN1CCCC12CN(C(C1CC=CCN1C(=O)C=CC(=O)NC1CC1)=O)C2 c1(NC(C2CCN(C(=O)NC(c3ncco3)C)C2)=O)ccccc1 C1(CC)(NC(C2CCC(O)CC2)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC1 C1(COC)CCN(C(C2CC23CCN(C(=O)CC2(O)CCC2)C3)=O)C1(C)C c1(CC)nc(C(N2CCC(O)(C(C)NC(C3(F)CCCC3)=O)C2)=O)c(C)o1 CCC(C)C(CO)CN=C(NCc1ccc(F)cc1)N1CCC(CC(F)(F)F)C1 CC1(C)C2CCC1(C(=O)NCCC(O)C(=O)NCCCc1cccnc1)C2 CON(CCC(=O)NC(c1ncc(C)[nH]1)(C)C)C(=O)C1CC1C C1(C(=O)NC2CC(CCC)C2)(COC)CCCN1C(=O)CC1CCCN(C)C1 C1(CNC(CN(C2CCCC2)C)=O)COCCN1C(=O)C(C1CCOCC1)=O N1(C(c2cc(CCC)n(C)n2)=O)CCCC2C1CCN2C(c1cncc(C)c1)=O CCCC(C)(CC)C(=O)N1CC(CCNC(c2ccc3cnnn3c2)=O)C1 N1(C(C(c2ccnn2C)C)=O)CCCCCCC1C(=O)NC1(CO)CCOC1 C1(C(N2CC(CNC(CC34CC(C(=O)OC)(C3)C4)=O)C2)=O)CC(C)(C)C(=O)C1 S(=O)(=O)(c1cc(C(=O)NCC2(O)CCN(C(=O)C(O)C(C)C)C2)co1)NC Cc1nc(N2CCC(c3cccc(F)n3)C2)c2cnn(CCO)c2n1 C1(C)(C(N(CCNC(Cn2ncc(CC)c2)=O)CCOCCO)=O)CC(C#N)C1 C1(NC(C(CSC)O)=O)C2CN(C(C3CCOC3c3ccc(Cl)cc3)=O)CC12 c1(C(=O)NC2CCC(NC(C(CC)C(C)O)=O)CC2)cccc2c1OC(F)(F)O2 Cc1cc(CC(N2CCC(Cc3nn[nH]n3)C2)=O)on1 C1(COC)CC(OC)CCN1c1nc(-c2ccncc2)ncc1C C1(C(=O)NCCN(C(=O)C2=CCCCO2)C)CCC2(CC1)NC(=O)N(C)C2=O C#CCC(O)C(=O)NCCCCNC(=O)Cc1cnc(C(F)(F)F)s1 c1(C(N2CCN(C(CCc3nc(C)c(C)o3)=O)CC2C)=O)ncnc2sccc12 N1(C(CC)=O)CC(CNC(=O)C(C(C)O)NC(=O)OC(C)(C)C)C(C)(C)C1 N1(C(C(CO)NC(C(CC)n2ccnc2)=O)=O)CC2CC=CC1C2 Cc1cc2[nH]c(C(N3CCCCC3CNC(=O)C(C3CC3)N(C)C)=O)cc2s1 N1(C(C2(CC)COC2)=O)CCCC(O)(CN(C(=O)CC2CCCS(=O)(=O)C2)C)C1 CCCC(CCCNC(=O)CCCNC(C)=O)NC(=O)C=CCn1cncn1 N1(C(c2c(C)nc(C)s2)=O)CC2CC(C1)CN(C(C1Cc3cccnc3C1)=O)C2 CCCC(C(O)C(=O)N1CC[Si](C)(C)C1)NC(c1ncsc1C)=O C1(CC(=O)N(c2cnn(C)c2)CC#C)CN(C(=O)CCCC(C)C)CC1C=C c1(C(OC)OC)cccc(CCNC(=O)CCC2CC2C(C)C)c1.CCS C1(CC(=O)NCC(COCC)(C)C)CC(O)CN1C(c1cscc1CC)=O N1(C(CC(=O)NC2CC2)=O)CCC2(CCC(NC(c3cc[nH]n3)=O)C2)C1 N1(CC(=O)NC(c2ccccc2F)CNC(C2(O)CCOC2)=O)CCCCC1=O c1(NC(C2C3CN(Cc4c(C)ccnc4)C2C3)=O)ccc([N+](=O)[O-])c(C)c1 C(=O)(CC(F)(F)CC)N(C(CC(=O)NCC1CN(CC)C(=O)O1)CC)C N1(CCN(C)C(C2(CCF)CCNC2)=O)CCCC(CN2CCNCC2)C1 N1(C(C(c2c(Cl)cccc2Cl)C)=O)CCN(C(c2c[nH]nc2F)=O)C2(CC2)C1 C(=O)(C1=CCCCCC1)NCCC1(NC(C2C(c3n(C)ncc3)C2)=O)CCC1 c1(C2CCN(C(N3CC(C)(C)OCC3)=O)CC2)ccc2ccccc2n1 c1(C(=O)NCCC2CC(OC)CN2C(=O)C=CC2CC2)cccc2oncc12 C1(C)(C(N(CC(C)(C)CNC(C2CC2C(C)(C)C)=O)C)=O)CC(C)(C)C1 c1(C(N2CC(CN(C(c3cnc(C(C)C)s3)=O)C)C2)=O)sc(F)cc1Cl c1(OC)ccc(CCNC(=O)C(=O)NCC2CCC(N)C2)cc1 N1(C(C2C(C)C2)=O)CC2C3CCC(C2C1)N(C(=O)Cc1cnn2c1CCCC2)C3 C(=O)(CCCCNC(=O)CCC1NC(=O)NC1=O)NC(C)CSC(F)F C1(C(N2C(c3n(C)ncn3)COCC2)=O)CCCC2(C1)CC(O)C2 C1(NC(CN(C(=O)C(C2CCC2)OC)CC)=O)CC(C)(C)O1 c1(C(c2n(CC=C)nnn2)NCC2(C3CC3)CCC2)c(Cl)ccc(F)c1Cl c1(CC)cc(C(=O)NCCC(O)CNC(c2ccsc2Cl)=O)ccc1Cl CCCC(O)CC(=O)NC1(CC)CCN(CC(O)COCCOCC)CC1 N1(C(C2(C(=O)OC)CC2)=O)CCC(C(=O)NC2CC2(C)C)=C(F)C1 c1(C(N2CCC(NC(C(C)=C(CC)C)=O)C(F)C2)=O)c(N)ccc(F)c1C C1(O)(CNC(=O)CC2CCCN(C(c3cc(CO)ccn3)=O)C2)CCCCCC1 c1(N2CC(NC(C(C)CC3CC3)=O)(CSc3ccccc3)C2)nc(Cl)c(C#N)s1 N1(C(CC(C)(C)c2cccs2)=O)CCC2(CCC2)C(NC(=O)CCC(C)(C)F)C1 Cc1[nH]nc(C(=O)Nc2ccc(CC(C)C)cc2)c1F c1(CNC2C3CN(C(c4ccnc(OC)c4F)=O)CC32)cc(I)c(C)c(I)c1 C1(NC(c2c(C)nn(CC(F)F)c2)=O)CCC(C)(CNC(c2csnn2)=O)CC1 C1(NC(C2CCCC2)=O)CN(C(c2c[nH]cc(Cl)c2=O)=O)CCC1CO C1(C2(NC(C(C)SC)=O)CC2)CCCN(C(=O)CC(C)n2ccnc2)C1 C12(COC)CC(CNC(=O)C(CCO)N(C)C)(CN1C(=O)CCC(=O)N(C)C)C2 N1(CNCc2nccc(C)n2)CC(C)OC(C)C1.C12(CC1)CC2.C(C)(C)(C)OC(=O)N c1(OC)c(CC(=O)NCC2CC(O)CN2C(=O)C(C)OC(C)(C)C)cccc1F c1(C(C(=O)NCC=C)N(CCCCC=C)C)ncccc1Br Cc1c(C(N2CC=CC(NC(c3coc(Cl)c3)=O)C2)=O)cnn1C1CCC1 c1(C(=O)NC(C(C)NC(c2ccc(C#N)s2)=O)CO)onc2c1CCCC2 c1(C(N2CC(O)(C(C)NC(=O)CC3(N4CCCC4)CC3)C2)=O)cnn2ccccc12 CN1CC2(CC2)CC1C(N1CCC(O)C1C(N1CCC1(C)CCO)=O)=O C1(O)(C(C)C)CCN(C(=O)C(C)(C)C2CCCN2C(=O)COCc2nc[nH]n2)C1 c1(CC(N2CC(NC(=O)CC3CCCCCCC3)C2)=O)cnc2c(=O)[nH]ccn12 C(=O)(CCS(=O)(=O)Cc1ccccc1)N(CCNC(=O)CCC1CCOC1)CC O=C(C1CCc2ccccc21)NC1C2CC1N(C(c1cscc1C(F)(F)F)=O)C2 C(=O)(C(C(C)C)N(C)C)NC1CC(CCNC(c2ccn(CCC)n2)=O)C1 c1(NC(C2CCNC2)=O)ccc(F)c(Nc2cc(-n3cncn3)ncn2)c1 C1(C(=O)Nc2onc(C)n2)CCN(N2CC(N(C)C)C(C)C2)CC1 C(=O)(C(C)(C)CC(F)F)NC1CN(C(C(C)OCCC=C)=O)CC(O)C1 C12(C(N(CC(CN(C(C(C)(C)OC)=O)C)O)C)=O)CC3CC(CC(C3)O1)C2 c1(C(=O)NC2C(N(C(C(C=C=C)C)=O)C)CCCC2)cc(C)cc([N+](=O)[O-])c1N c1(CSC)ccc(OCCNCc2c(C(=O)OC)c[nH]n2)cc1OC CC(C)(C)C(C(=O)NC1(CN(C)C(C2(CN(C)C)CC2)=O)CC1)C(O)C(F)(F)F C1(C(=O)N(CCC2CC2)CC)CCC(CNC(c2cc(CC)on2)=O)CC1.C1(C)CC1 CC1COc2c(C(=O)NC3CC3CNC(c3snnc3C3CC3)=O)cnn2C1 C(=O)(C(C)S(N)(=O)=O)N1C(C(=O)NCC2CN3CCC2CC3)(COC)C=CC1 N1(C(c2ncn(CC)c2)=O)CCC(C)CC1C(=O)NCC1(CC)CCOC1 n1(CC(=O)NC2CC2(c2ccccc2)C)c(=O)ccc2ccccc12 c1(OC)ccc(CN2CCSCC2C(=O)Nc2ncccc2Br)c(Cl)c1 c1(N(C2(C#C)CCCC2)C)nc2cc[nH]c2c(=NC(C)c2ccc(C#C)cc2)[nH]1 c1(C(N2CC3CCC2CN3C(C2CCC2)=O)=O)cc(F)ccc1[N+](=O)[O-] C=CCCC(F)(F)C(=O)NC1CC(F)(CNC(=O)Cc2cc(F)ccc2Cl)C1 CCC(C)(C)CC(=O)NCc1cc(C(=O)NCCc2cn[nH]c2)on1 C1(C(=O)NCCC2(CNC(=O)CC3OCCO3)CC2)COc2ccc(Cl)cc2C1 C(c1c(C)nn(CCC)c1Cl)=CC(N1CC(NC(C2(CC#C)CC2)=O)C(C)C1)=O Cc1cc(Cl)c(CC(N2CCN(C(=O)CCC(F)(F)F)C(C3CC3)C2)=O)cn1 c1(C(N2CC(CNC(C=C(C)Cl)=O)C(C)C2)=O)nc(C)ncc1Cl C1(C(=O)NC(C)C(=O)NCc2ccc(C3CC3)o2)COC(=O)N1 c1(C(CO)N(C(C2(CC)CC(C)(C)C2)C(=O)O)C)ccc(F)c(C)c1 C1(C(N(CC(=O)NC(C2CC23CCC3)C2CC2)CC)=O)C2CCC(C2)C1C c1(C(=O)NC23CC(CNC(C45C(C)(C)OCC4C5)=O)(C2)C3)nc2ccccn2n1 C1(CNC(C(C)OCCCC)=O)CCC(CC(=O)NC2(C)CS(=O)(=O)C2)CC1 C1(NC(c2cn(C)nc2-c2ccccc2)=O)CN(Cc2ccccc2)C(C)(C)C1 c1(C(=O)NCCC2CCCN(c3cnc(F)cn3)C2)cc2c(nc1O)CCC2 C1(C(=O)NC2C3CN(C(C(CN(C)C)O)=O)CC32)CCC2(CC1)CC2 C(=O)(CCCCC(F)(F)F)N(C)CC1CCCC1NC(=O)CCCCC CC1CN2CC1N=C1NC3=C(C(=NC4CC5CC2CC45)N1)COCC3 C12(C(N3CC(NC(C4OCC(C)C4)=O)C(C)C3)=O)CCCC(C)(C1)OC2 c1(N(C(=O)NC(C#C)(C)C2CC2)C)cc(COC)ccc1Br N1(C(=O)CSCc2nccs2)C2C=C(c3ccccc3)CC1CC2 C=CC(C)(C)CCCNC(=O)C(C)(C1CC1)N(C(=O)CCCCSC)C C(C(COC)CC(=O)NCC(C)N(C(=O)C(C)NC(=O)C=CCl)C)OC C(C(C(=O)NCCCCN(C(=O)CCC1CCC1)C)N(C)C)N(C)C C1(C)(C(=O)OC2CN(C(C(C)Sc3ncccn3)=O)C2)CCC(=O)CC1 N1(C(C(F)OC)=O)CCC(C)(CNC(=O)COCc2ccnc(O)c2)C1 C1(C(c2nnnn2C)NC(CCC)C)(OCC)CCC2(CC1)COC2 Cc1cncc(CC(=O)NCC2(F)CCN(C(=O)Cc3cc(C)oc3C)C2)c1 Cc1cn2cc(C(=O)N(C(C)CN(C)C(c3cc(N)cc(F)c3)=O)C)ccc2n1 CCC(C)C(=O)C(=O)N1CC(Cn2cc(-c3cnn(C)c3COC(C)C)nn2)C1 N1(C(C(C)NC=O)=O)CCn2nc(C(=O)N(c3cccc(O)c3)CC#N)cc2C1 c1(C(N2C(C)CC(CNC(c3c(C)cccn3)=O)C2)=O)ccc(F)c(O)c1 c1(C(=O)NCc2cccc(CN(C(=O)CSC3CC3)C)c2)cnn(C)c1Cl c1(CC)[nH]nc(C(N2CCC2C(=O)Nc2ncccc2C)=O)c1F N1(C(C2CCN(C(c3cc(Cl)cc(Cl)c3)=O)C2)=O)CCN2CC(O)CC2C1 c1(NC(C)CCNC(=O)C(C)(O)c2ccccc2)cc(C2CCC2)ncn1 c1(OC)cc(N)c(C(N2CC(O)CC23CNC3)=O)cc1Br.C12=CC=C(C=C1)C2 C(CCC(=O)NCC(c1ccccc1)NC(c1nn[nH]c1Cl)=O)OCCC C1(C(N(C2CCCN(C(=O)C(F)n3cccn3)CC2)C)=O)CCCCS1(=O)=O CC(C)C(CN(C)C)C(=O)N1CCC(CO)(CNC(=O)CC2CCSC2)CC1 c1(C(N2C(c3cn(-c4cnn(C)c4Br)nn3)CCC2)=O)ccc2ccccc2n1 O(C1(OCC)c2cccnc2COC1(C)C)CC(=O)NC1C(C=C)CC1 CC1CC(C(N2CCC(O)(C(N)=O)CC2)=O)CN(C(c2cnn(C)c2)=O)C1 C1(CNC(c2cnccc2Cl)=O)CN(C(c2nc(C3CC3)cs2)=O)CC12CC2 C1(N(C)C(c2cncc(F)c2)=O)CCC(NC(=O)CC23CCCC2C3)CC1 Cc1ccc(=NCCC(=O)N(C)CCNC(C2CC(OC)C(N(C)C)C2)=O)[nH]c1 c1(C2(C(=O)NCCNC(=O)C(F)C3CCC3)COC2)ccccc1 c1(OC)cnc(Cl)nc1N1CCCC(C)(CNC(c2cc(C)c(C)s2)=O)C1 CC(C)C(C(=O)NC(=O)NC1(C)CN(c2ccccc2)C1)NCc1ccccc1 CC1CCCN(CC(=O)Nc2ccc(C(F)(F)C(F)F)cc2)C1CC(N)=O C1(NC(C(c2c(OC)cccc2)C)=O)CCN(C(c2cncc(F)c2)=O)CC1O C1(CNC(=O)CCc2cccnc2)CN(C(c2nncs2)=O)C2(CCC2)C1 C1(C(N(CCC(=O)NC2CCCC2C2CC2)C)=O)CCCCN1C C#CCC(CC#C)C(=O)N1CCN(C(c2cccc(O)n2)=O)C(CCO)C1 C(=O)(CCCn1nnnc1C1C=CC(NCC(C)(C)N(C)C)C1)OCC CN1CCOC(C(=O)N(C2CC2)CC2COCCN2C(=O)CCn2cccn2)C1 N1(C(c2cn(C)nc2O)=O)CCCN(CCNC(=O)CCN2CCCC2)CC1 C(=O)(C(C)(C)C(=O)NCc1cncc(C(=O)NOCC(C)C)c1)OCC Cc1ccc(C(N2CCCC(CCNC(C3CCC(=O)N3)=O)C2)=O)c(C2CC2)c1 N1(C(CC(=O)NCC)=O)CCCC(C)(C)C1CNC(c1ccc(N)cc1OC)=O C1(CCNC(C(C=C)O)=O)CSCCN1C(c1cc[nH]c(=N)c1)=O c1(C(=O)NCC2N(C(CCC(=O)OC(C)(C)C)=O)CCCC2)ccc(F)cc1F c1(CC)cc(F)ccc1C(N1CC(CCNC(=O)CC(F)(F)Cl)OC(C)C1)=O c1(OCc2ccc(OCc3cc(C)c(O)cc3)cc2)ncnc2cc(Br)cnc12 C12(NC(c3cnn(C)n3)=O)CCCC1CN(C(c1csc(C#N)c1)=O)C2 C1(C)(NC(c2cnc(COC)s2)=O)CCN(C(c2cccc[n+]2[O-])=O)C1 C1(NC(c2ccn3ccnc3n2)=O)CCC2CN(C(=O)Nc3cn[nH]c3)CCC2C1 C1(N(C)C(C2CC(=O)N(C(C)(C)C)C2)=O)CN(C(=O)Cn2cccc2)CC1(C)C N1(C(COC)=O)CC2CCC2(CCNC(C2(Cl)CC23CCC3)=O)C1 c1(C(N2CC(CC)C(NC(c3ccoc3C)=O)C2)=O)cc2nc(Cl)ccc2o1 c1(C(=O)OC)cc(C(c2nnnn2C)NCc2ncsn2)[nH]n1 c1(C(N2CCCC(NC(C(C)C)=O)C2C)=O)ccc(C(F)(F)F)c(Cl)c1Cl N1(C(C(C)(F)F)=O)CCC2(CCC(CNC(c3ccnnc3S)=O)OC2)CC1 Cc1cc(C(=O)NCCCCN(C)C(C2(C)CCCNC2=O)=O)cc2c1CCC2 C1(NC(c2scc(C(N)=O)c2)=O)CC(NC(C2CCC(=O)NC2)=O)C(O)C1 CC(c1cccc(Cl)c1)=CC(=O)NCC(c1ccccc1)Oc1ccccc1 C1(C(=O)NC2CC2)CCN(C(=O)CCOCC2CC2)C12CCC2 N1(C(CC=C=C)=O)CCN(C(C2CC(C)(C)CCO2)=O)C(CC)C1 c1(NC(C2CN(c3ccc(F)cc3)C(=O)C2)=O)nccc(Cl)c1I c1(NC(c2ccccc2-n2cccn2)=O)cc(Cl)ccc1CO c1(C(=O)NC(c2cn(CCC3CCCC(C)C3)nn2)C)csc2ccc(I)cc12 N1(C(CC(C)(C)C#N)=O)CCCC2(C1)CN(C(c1ncc(Br)cc1O)=O)C2 n1(CCCCC)c(N2CCOC(c3cccc(Cl)c3)C2)nnc1COCCCC N1(C(CSC)=O)CC2(CCN(C(C3CCC(C(C)(C)O)CC3)=O)C2)C1 C(=O)(C(C(=O)N1CCC(CO)(CNC(=O)CN2CC3CC3C2)CC1)C(C)C)OCC c1(C(=O)NC(C2CCN(C(=O)CCc3ccoc3)CC2)C)ccnc(CO)c1 C(=O)(C(C(C)O)N(C)C)NC1C(C(=O)NC(CCC=C)C)COC1 c1(OC)cc(C(=O)NCCC2CC(NC(=O)C#CC3CC3)C2)c(Br)c(F)c1 c1(C(=O)NC2(C(=O)NC(C#CC)(C)C)CC2(C)C)c(C)noc1C C(=O)(C#CC1CCOCC1)N1CC(C)C(CNC(c2ncc3n2CCCC3)=O)C1 O(N=C1CCCCCC1)CC(N1CCC(C)(NC(c2ccsc2C#N)=O)C1)=O C(=O)(CCCC(F)(F)F)NCC(C1CC1)NC(c1ccc(C(CC)C)cc1)=O C(=O)(C(CC)C(F)(F)F)N1CC(N(C(CCC#C)=O)C)C2(C1)CC2 C1(C(N2CCC(N(C)C(C3CC4CCC(C3)O4)=O)C2)=O)CCC2(CC1)CC2(F)F N1(C(C)C(=O)NCCNC(C2(C)CC2(C)C)=O)C(=O)CCC1=O c1(C(N2C(CC(=O)NC3(CSC)CC3)CC(C)(C)C2)=O)cc(C#N)ccc1N Cc1ncc(Br)cc1C(=O)NCCC1(O)CCCN(C(C2(O)CCC2)=O)C1 c1(OCC)cc(CN2CCOCC2(C)CC)cc2c1OCCO2 c1(C(C(F)(F)F)C(=O)NCC(N2CCOC2=O)(C)C)cc(Cl)cc(Cl)c1 Cc1c(C(N2CCN(C(C3CCC(=O)NC3)=O)CC(O)C2)=O)cnc2ncnn12 C(=O)(CC1=CCN(C(=O)C(C)(O)C2CC2)CC1)NC1CC(C)SC1 Cc1cc(C(=O)NC2CCCN(C(c3csc(O)n3)=O)C2C)cc(C)c1F C1(CC)CN(C(c2cnc(F)c(Cl)c2)=O)CCC1N=c1cc(C)nc(OC)[nH]1 c1(C(N2CCN(C)CC2CNC(c2ccc(Cl)cc2)=O)=O)cc([N+](=O)[O-])nn1C C(=O)(CCC1CCc2ccccc21)N1CC(NC(=O)CCC2CCC2)C2(C1)CC2 N1(C(C(c2cncnc2)C)=O)CC(C2CCN(C(c3ncncc3N)=O)CC2)C1 Cc1ccc2ncn(CC(=O)N(C3CN(C(c4ccnc(S)c4)=O)C3)C)c2c1 c1(C(N(CCNC(CN(CCOC)C)=O)C)=O)cc2sc(S(N)(=O)=O)cc2s1 c1(C(N(CCCNC(C2(N(C)C)CCC2)=O)C(C)C)=O)cc2cccc(F)c2o1 C1(c2n(CCOC)nnn2)(NC(C)CCCC(C)C)COC2(CCC2)C1 C(=O)(CCC(C)S(C)(=O)=O)NC1CCCN(C(CC=C(C)C)=O)CC1 CC(C(=O)NC12CCCN(C(c3ccc(NC=O)cc3)=O)CC1C2)C1=CCCC1 Cc1cnc(Br)cc1NC(=O)CCCn1cc(-c2cnc(Br)nc2)nn1 c1(C(=O)NCC2CN(C3CCCC3)CCO2)cc2c(s1)CCCCC2 N(C(=NCCCF)NCC1CCN(S(C)(=O)=O)C1)CC(C(C)(C)C)SC C1(C)(NC(C2(CNC(CC(C)OC)=O)CC2)=O)CCCC1(C)C C(c1nccs1)=CC(=O)NC(C(=O)NCC1(O)CCSC1)c1cccs1 Cc1cc(C(=O)NC(C)(C)CC(=O)NCC(C)C(C)(F)F)ccn1 C(=O)(CCCC(F)(F)F)NCC12CCC(NC(C=Cc3scc(C)n3)=O)(C1)CO2 CC(C)C(CCNC(=O)CC(C)C1CC1)N(C(=O)CSCc1cccs1)C c1(C(C)C)cccc(C(=O)NCCN(C(=O)CC(C)n2cccn2)CCOC)n1 c1(NC(N2CCC(F)C2)=O)cnc2c(c1)CN(Cc1cc(F)ccn1)CC2 c1(C(c2nnnn2CCSC)NC(C=C)(C)C)csc(CC)n1 Cc1ccc(C(=O)NC(C)(C)C(=O)N(C2CC2)CC2CCOC2)o1 CN1CCN(C(C2CCC(C(N)=O)C2)=O)CC1CNC(C1C2CC3C(C2)C13)=O CCCCCC(O)C(C)C(=O)NCC1CC(NC(C2(C3CC3)CC2)=O)C1 CCCCN=C(NCCCOC1CCCCC1)NC1CCCSC1 N1(C(Cc2c(C)scc2)=O)CCN(C)CC1C(=O)N(C)Cc1ccns1 C(CCC(=O)NC1CC(CNC(=O)C(C)(C)n2ccnn2)C1)N(C(C)=O)C CCCC(CCC)C(=O)N1CCN(C(c2cnsc2)=O)CC(C)C1 c1(SC)ccc(C=CC(=O)NCCCC(C)NC(=O)CN(C)CCO)cc1 C=CCC(CC=C)CS(=O)(=O)N1CCC2CCCCC12 C1(CC(=O)NCC(C)(C)OCC(=O)NCC2(N(C)C)CC2)CCCCO1 C1(C)(CNC(CCSCCC)=O)CCCN(C(=O)C(CCOC)OC)C1 N1(C(CC(=O)OC)=O)CCCC(CCNC(=O)CC2CCCN2C(C)C)C1 N1(C(c2ccc(F)s2)=O)CCC2(CCCN2C(=O)Cc2cccc(F)c2)C1 N1(C(COC)=O)CC2CC(N(C(=O)C(C(C)C)c3cccnc3)C)C1C2 C12(C(=O)NCC3CCC(C(=O)NCCC(C)(C)O)CC3)CCC(CC1)CO2 c1(C(=O)NC2CC(F)(C(=O)O)C2)nsnc1O N1(C(c2scc(C(N)=O)c2)=O)C2CCC1C(CNC(=O)CNC(=O)C1CC1)C2 Cc1cc(N)c(C(=O)NC2CCC3CC23)cc1C C1(CNC(c2on(C)c(=O)c2)=O)CC2CCC1N(C(=O)COC1CCCOC1)C2 N1(C(C#C)=O)CCC2(CC2C(=O)NC2(C(F)(F)F)CC2)C1 C(=O)(C(O)CCC(C)C)N(CCCNC(C1C(C)(C(=O)OCC)C1)=O)C1CC1 CC1=CCC(C(=O)N(C(C)C(=O)NCc2cc(C)nn2C)C)CC1 c1(C(=O)NC2CN(C(C3CC34CC(O)C4)=O)CCC2O)cccc2c1CCC2 c1(-c2cncc(CC)c2)ccc2c(C(=O)N(C)CC3CCCCC3)c[nH]c2c1 C(=O)(C(CNC(c1cnn(C(C)C)n1)=O)C(C)C)N(CCCO)CCC C1(NC(C(C)CF)=O)CN(C(=O)C(CC(N)=O)c2ccc(F)cc2)C2(CCC2)C1 C(C(C(F)(F)F)N1CCN(C(=O)CNc2cn[nH]c2)CC1)NC(C=CCC)=O c1(OC)cccc(NC(=O)CC2(CC(=O)C(F)(F)c3cnnn3C)CC2)c1C CCC(CCCC(=O)NCCCc1ncn(C)n1)NC(C1(O)CCCC1)=O N1(C(c2ccc(C)cc2Cl)C(=O)NCC(F)F)CCC(C2CCCC2)C1 N1(C(CSC(C)C)=O)CCC(C)(C)C1CNC(=O)COc1ccc(F)c(F)c1 CCCCCCCC(=O)N1CCN(C(c2ccc(O)nn2)=O)C2CC12 C1(NC(C(CSC)O)=O)CN(C(=O)CCCCc2ccc(F)cc2)CC(F)(F)C1 CCCCCCCCCC(=O)N1CCCC(CNC(=O)C(F)CC(C)C)C1 O=C1CCCC(C(=O)NC2(C(=O)NCC3COC(=O)N3)CCCCC2)N1 C=C1CC2(C1)CC(C(N1CCN(C(=O)CCN3CCC(C)CC3)C(CO)C1)=O)C2 c1(C2(CN(C(=O)Cn3cccn3)CCn3cccn3)CC2)ccc(C(=O)O)cc1 CC(c1ccco1)=CC(=O)NCCCOCCN(c1ccnc(C2CC2)n1)C C1(O)(CNC(CCOCCOC)=O)CCCN(C(=O)COc2cccc(C)c2)C1 c1(CC(=O)Nc2cccc(C(N3CC4CCCC4C3)=O)c2)ccc(O)c(Br)c1 CC1(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CC(C(N)=O)C2(C)C)=O)CC1 C1(C(=O)NC(c2cccnc2)CC)CCCN1NC(=O)C(C)(C)COC c1(CN(C)CCCCNC(=O)NC(N)=O)ccnn1-c1ccccc1 C1(NC(C(C)N(C)C)=O)CCCC1NC(=O)CCCc1ccccn1 C(=O)(C1=CCCOC1)N1CC(CCC)C(C(N2CCC3CC23)=O)C1 N1(C(C(C(=O)OCC)OC)=O)CCC(C(=O)NCC(CC)CCO)C12CCC2 c1(C2(C)CC2)cc(C(=O)NCCC23CC(NC(=O)CNC=O)(C2)C3)no1 CCCC(C)(C)CC(=O)NC12CCC(NC(C3CC(C4CC4)=NO3)=O)(CC1)C2 c1(C(=O)NCC=CCNC(CC2(C)CCCCC2)=O)ccc(C2CC2)c(Cl)c1 C12(NC(=O)CC3CCCC3)CCCCC1CN(C(c1cnc3n1CCS3)=O)C2 C1(C2CCC2)(C(N2CC(O)CC(NC(c3c(C)nncc3)=O)C2)=O)CC1(F)F CC#CCCC(=O)NC1(CCO)CN(C(c2cccc(C(F)(F)F)n2)=O)C1 CC(C)CC(Cc1ccccc1)C(=O)NCCC(C)NC(c1ncncc1F)=O c1(C(N2CCC(OCCNC(C3CC=CCO3)=O)C2)=O)cccc(=O)n1O C1(C(N2CCC3C(NC(c4ccc5nonc5c4)=O)C32)=O)CC2(C1)CC(F)(F)C2 C1(C)(COC)CC(NC(c2coc(C)n2)=O)CN1C(=O)C(CN(C)C)N(C)C C(=O)(C1CCCn2nccc21)NCCC(C)Nc1nccc(C)n1 CC1(C)C(NC(C2CCCCN2N=O)=O)CCN1C(c1csnc1Cl)=O N1(C(Cc2cncc(C)c2)=O)CCC2C(NC(=O)CCCCCNC(N)=O)CC12 N1(C(C(=O)NCC)=O)CCN(C(=O)C(=O)C(C)(C)C)CCC1C c12ccc(cc1Cl)NC(=O)C(=O)N2.C(c1ccco1)=CC(=O)OC(C)(C)C N#Cc1cc(CN(C2CN(C(=O)Nc3ccc(Cl)cc3)C2)C)ccc1Cl N1(CC)CCOC(C(=O)NCC(F)CNC(=O)CCC(=O)c2cccc(N)c2)C1 C(C(C)(O)CC(=O)N1CCN(C(c2cnc(C(F)F)s2)=O)CC1C1CC1)OC CC(C)(CO)C(C=Cc1ccccc1)NC(=O)Nc1ccccc1Cl C(=O)(C(C)C(C)n1cccn1)NCC1C(NC(CSCCCC)=O)COC1 C1(C(N2CCCCC(N(C)C(C3CCCCC3O)=O)C2)=O)CC2CCC1C21CC1 C1(NC(C2CCCC2)=O)CCOC12CCN(c1nnc(C(F)(F)F)s1)CC2 c1(C(=O)NCCCNC(CSC(=N)N)=O)cccnc1CN1CCSCC1 CCC(CCC(=O)N(C)CCc1cccs1)NC(=O)CN1CC(OC)C1 c1(C(N(C)CC2N(C(CNC(=O)OC)=O)CC(F)C2)=O)cc(N)cc(F)c1 c1(C(C)NC(C2(F)CCN(C(c3ccns3)=O)C2)=O)ccc2c(c1)CCC2 Cc1cc(C(=O)NCCNC(c2nc(OCc3ccccc3)c(C)s2)=O)n(C)n1 N1(C(c2cncc(CC)c2)=O)CCC(C2(NC(C3CCCC3C(F)F)=O)CC2)C1 C(N=c1cc[nH]cc1S(=O)(=O)NCC1CCCO1)C1(OC)CCSC1 CN1CCC(CC(N2CC(OCCNC(C3CC4CC4C3)=O)C2)=O)CC1 Cn1ncc(C#N)c1C(N1CC2CC(NC(c3ccc(F)c(F)c3)=O)C1C2)=O N1(Cc2c(OC(F)F)ccc(C)c2)CCC(C2CCCOC2)CC1 n1(CC)nnc2cc(C(N3CCC(C)N(C(=O)COCC(F)F)CC3)=O)ccc12 N#Cc1cc(NNCc2cccc(CS(N)(=O)=O)c2)ccc1Br C(C)(CNC(=O)CC1C=CS(=O)(=O)C1)(C(C)C)NC(CCC=C)=O Cc1cc(C)cc(C=CC(N2CCC3CC2CN3C(C2CC23CC3)=O)=O)c1 C1(NC(CCC(C)OCC)=O)C2CCC1N(C(C1(OC)CCCCCC1)=O)C2 C1(NC(CC(COC)(C)C)=O)COC2(C1)CN(c1ncnc(Cl)c1C(=O)OC)C2 N1(C(C(C(C)C(F)(F)F)F)=O)CCCC2(CCN(C(c3cccn3C)=O)CC2)C1 C=C(C)CC(C)C(=O)N1CC(NC(c2cc(NC(C)=O)ccc2N)=O)C2(CC2)C1 c1(C(C(=O)NCCOCCCN(C)C(c2cn(C)nc2O)=O)F)ccc(F)cc1 CC1CCCc2cc(C(N3CC(NC(c4cn(C)nn4)=O)C(F)C3)=O)nn21 c1(OC)ccc(C(=O)NCC(C)(C)NC(c2nccnc2N)=O)c(OC(C)C)c1 Cc1cc(Cl)c(C(N2CCC(CC(C)NC(c3ncoc3C)=O)CC2)=O)cn1 N1(C(C2N(C)CCN(C)C2)=O)CCC2C(CCCN2C(=O)C=CCO)C1 c1(C(N2CC(C)S(=O)CC2)=O)cc2cncc(Br)c2s1 C12CCN(CC1(C)C)C(=O)c1ncc(s1)C(=O)N2.C1(C(C)(C)OC)(COCC)CC1 c1(C(=O)NC2CN(C(C(C(C)C)C#N)=O)C(C)CC2)cncc2sccc12 c1(-n2cc(C(=O)NCCCOCc3nscc3Br)nn2)ccccc1Cl CC1CCC(NC(=O)CC23CCC(C)(C2)OC3)CN1C(c1cc2scnc2[nH]1)=O c1(C(N2C(C)CC(NC(CCCOCCOC)=O)C2)=O)cnc2[nH]ccc2n1 N1(c2nnc(CC)n2CCCCC(c2ccccc2)(C)C)CCOC(C)C1(C)C C(CNC(c1c[nH]c(=N)o1)=O)(C(=O)NCC(C)CC1CC1)OC C1(CC(=O)NCC(CC)(C)CO)N(C(c2cc(O)nn2C)=O)CCC1(C)C c1(C(=O)NC(CNC(c2cnn3c2NCCC3)=O)C2CC2)cnc2[nH]nnc2c1 C1(NC2(C(=O)OC)CCCC2)C(C)CCCN1C(=O)CCc1ccccc1F c1(OC)ccc2[nH]c(C(=O)NC3CC3C(=O)NCCC(C)(C)O)cc2n1 c1(C(=O)NC(CNC(CC2ON=C(CC)C2)=O)C)nccn2ccnc12 C1(NC(C2C(COC)CC2)=O)CCC(O)CN(C(C2CC23CCCC3)=O)C1 c1(C(=O)NC(CNC(c2ccc(C(F)F)s2)=O)C2CC2)nccc2occc12 N1(C(C(CC)C(=O)OC)=O)CCOC2(C1)CN(C(c1cc(C)sc1C)=O)C2 Cc1cc(C(N2CCC(CCNC(=O)CSc3cnn(C)c3)CC2)=O)nc(O)c1 C1(C(=O)NCCCN(C(C2CC(CC)C2)=O)C)Cc2cc(C)ccc2O1 N1(C(c2ccn(C)c2)=O)CCC2(CCCC2NC(=O)COc2ccc(Cl)cc2)C1 CCCCCC(C)CC(=O)N(C)CC1CN(C(C2CCOC(CC)C2)=O)C1 N1(C(c2cnc(C(C)C)s2)=O)CC2CC1CCC2NC(=O)COc1cnn(C)c1 c1(C(=O)NC2(CCCNC(C(C)SC)=O)CC2)ccccc1-n1cccn1.C1(S)CC1 c1(C(=O)OC)cncn1CC(=O)NC1CC(CNC(=O)C=CCF)C1 c1(CC(=O)NCC2N(C(CCOC)=O)CC(C)C2)ccc([N+](=O)[O-])c(N)c1 N1(C(CCOCC#C)=O)CCN(CC2CCCN(C(c3cnn(C)n3)=O)C2)CC1 C1(NC(C2CC2F)=O)CC(F)CN(C(c2cc(F)cc(Br)c2)=O)C1 c1(CNC(c2cccc([N+](=O)[O-])c2)CC(=O)OC)cc(F)c(Br)cc1F C(=O)(C1=C(F)CN(C(=O)CCC2CC2(F)F)CC1)NC(CC)C1CCC1 CC1CC(C2CN(N3CCC4(CCCOC4)N3CC[SH](=O)=O)C2)=NO1 N1(C(C(CCC)C)=O)CC(NC(c2ccc(O)c(Cl)c2)=O)CC(C)C1 c1(Cn2cc(-c3cc(C)oc3)nn2)cnc(F)cc1C N1(CC(=O)NCCC2CC2)CCN(C(C2C3COCC23)=O)CC1 C(N=c1[nH]c(Cl)ncc1F)C1C(NC(c2c(C)nccn2)=O)CCCC1 c1(CC(=O)NC(C2OCCN(C(CC=C)=O)C2)C)ccc(S(=O)(=O)N(C)C)cc1 Cc1cccc2cc(C(N3CC(CO)(NC(C4CCNC4=O)=O)C3)=O)nn12 CC(C)(C(=O)N1CCC(NC(c2csc(C3CC3)c2)=O)C1)C1CCCO1 C1(OC(C(C2CCOCC2)OC)=O)(Cc2ccc(C(=O)OC)s2)CC(F)(F)C1 c1(C(=O)NCC2CC(NC(C3CC34CC4)=O)C2)nc(N2CCOCC2)ncc1Cl C1(C(=O)NC2(C)CC2)CCC2(CC2)CO1.c12cc(C)c(o1)C(=O)NC2.C(=O)(NC)N.C N1(C(C2CCN(C(=O)C3CC(O)(CC#C)C3)O2)=O)CC2CCC1C(O)C2 N1(C(C(C=CCCC)O)=O)CCC(C)(C)C(NC(=O)C(C)N(C)C(C)=O)C1 C1(F)(C(N(C(C)C)CC#N)=O)CCCN(C(C2CC2(F)F)=O)C1 C1(NC(=O)C(C)(C)C)CCC2CCCC1O2.C1(=O)CNC(=O)C2C(C2)C(C)N1 N1(C(c2cc(CCC)on2)=O)CCC(C)(CNC(C2(C3CCCCO3)CCC2)=O)C1 c1(CC)nnc2n1CCCC2C(=O)N1CCC(F)C(NC(c2ncsc2C)=O)C1 CCCC(C)(CCC)C(=O)NC(C1CCN(C(c2cc(C)nnc2O)=O)C1)C C1(CC#C)(C(=O)O)CCOC1.c12snnc1CC1CN(C1)C2=O.OC Cn1ccnc1CCC(=O)NCCC1(NC(c2cc(F)cs2)=O)CCCC1 C(CC(F)F)(C(=O)N1CC(C#N)(CCF)C1)N(C(C1N(C)CC1)=O)C1CC1 C(CC(=O)N1CCC(C(=O)NC(C2(O)CCC2)(C)C)O1)OC(C)=O N12CC3C(C3C1)CC(=O)NCCSCC2=O.C(C)(CNS(C)(=O)=O)OC C1(C(C)C)OCCC1C(=O)NCCCCNC(c1cc(C2CC2)no1)=O C1(CNC(C(C)C2CC2)=O)CC(=O)N(C2CN(C(=O)CC3CC(F)(F)C3)C2)C1 c1(N2CCC(NC(=O)NC3CC4(CCC4)C3)(CF)C2)ccc(F)cc1[N+](=O)[O-] CCCC(CC)CCC(=O)NC1CN(C(c2cc(N)cnc2Cl)=O)C1 c1(NCC2(NC(C(n3ccc(Br)n3)C)=O)CCC2)c(C#N)cccc1[N+](=O)[O-] C(=O)(C(F)C(C)(C)O)NCc1ccc(C(N(CC(C)(O)C)C2CC2)=O)o1 C(=O)(C1=NOC(C)(C)C1)NC(CNC(C1(C#C)CCOCC1)=O)(C)CO CC(C)C(C(=O)NCC1CCCCCN1C(=O)COCc1nccn1C)C(C)C C1(CNC(CCN(C(CC(CC)OC)=O)CC)=O)CCCC(C#N)C1 C1(C(N(C)CC2CCCN(C(c3ccc(COC)o3)=O)C2)=O)CC12CCCCC2 N1(C(C)C)CCCC1C(=O)N(C(CN(C(=O)CC1(C(F)(F)F)CC1)C(C)C)C1CC1)C CON(CCC(=O)N1CCOCC1C)C(=O)CN(C)C c1(CC)nc(C)c(C(N2CC=CC2CNC(=O)C(C)(F)CC)=O)s1 c1(NC(C2C(NC(CCC#C)=O)COC2)=O)cccc(Cl)c1 c1(C(=O)NC2C(CC)N(C(c3nc(C)sc3C)=O)CC2)nccn2nccc12 C1(C(N(C2CC(Nc3cc(O)nc(=O)n3C)C2)C)=O)Cc2ccccc2O1 C(=O)(CC1CCCc2ccccc21)NCC1CN(C(c2c(C)nn(C)c2F)=O)C1 CC1=C(C(=O)NC(C)CC2CN(C(c3cc(C)c(N)cn3)=O)C2)CCC1 C1(CC(=O)NCC(=C)F)CC2(CC2)CN1C(=O)CCC1CCC(C)O1 C(=O)(C(C(C)C)C(C)C)NC1CN(C(c2cnc(OC)c(C)n2)=O)C(CO)C1 Cc1cc(NC(C2CC(O)CN2C(c2cccc(F)c2I)=O)=O)ccc1Br C1(C(=O)NCC2(CNC(C(C)OCC)=O)CC2)C2CCC1C(F)(F)C2 C12(NC(c3nc(C)oc3)=O)CCCC1N(C(c1[nH]nnc1C1CC1)=O)CC2 C1(C(N2C(CC#C)CCCC2)=O)CN(C(c2nccn2C)=O)CC(C)(C)C1 N1(C(CC(=O)N(C)C)=O)CC(O)CCC1C(=O)NCCC1(C)CCOC1 C1(C(=O)NC2(CCNC(C3(C(N)=O)CC3)=O)CC2)CCCN(C(=O)C2CC2)C1 c1(C(=O)NC23CC(CNC(C(CSC)O)=O)(C2)OC3C)cccn2cc(C)nc12 c1(C(=O)NCc2cn(-c3ccc(OC)cc3)nn2)c(C)ccc(F)c1O c1(C(=O)NC2C(C)(C)C(C(=O)NCC3(CCO)CC3)C2)ccc2c(c1)CCC2 C(C(C)(CC(C)C)NC(=O)CC12CCC(CC1)C2)NC(C(CC)OC)=O c1(CC(N2CC(C)C(NC(=O)C(F)(F)C3CC3)CC2)=O)cccc2ccsc12 C1(NC(Cc2cnc(C)o2)=O)CCN(C(=O)CC(=O)NCC2CC2)C12CCC2 c1(OCC(=O)NC2CCC(CNC(C(CCOC)OC)=O)C2)ccc(Cl)cc1C S(=O)(=O)(c1ccc(C(=O)NCc2ccc3c(c2)OC(F)(F)O3)cc1)N(C(C)C)C c1(NC(C(C(=O)OCC)(F)F)=O)nc2cc(S(N)(=O)=O)ccc2o1 O=C1CC(NC(C2CC3CC2CC3NC(C2CN3CCC2CC3)=O)=O)CC(=O)N1 c1(NC(=O)C(c2cscn2)NC(C2CC3CCC2C3)=O)cccc(CO)c1.C1CC1 C1(C(=O)NCC2(OC)CN(C(c3csc(S)n3)=O)C2)CC2C=CC1CC2 Cc1cccc2[nH]cc(CN3CC(C(=O)NCC(C)(C)C)C(C)C3)c12 C1(CC)CC2CCC(C1)N2C(C1(C)CN(C(=O)C(F)OC(F)(F)F)C(C)(C)C1)=O N1(C(C=CC(CC)C)=O)CC2(CCC(CNC(c3noc4c3COCC4)=O)O2)C1 c1(CC(=O)NCC(C(C)C)NC(C2CCCC(=O)CC2)=O)ccc(F)c(Cl)c1F CC1(C)CCOC1CC(N1CCC(NC(c2cccnn2)=O)C1)=O c1(SCc2cccc(OC(C)C(=O)O)c2)ccc(Cl)cc1F c1(CC)[nH]nc(C(=O)N(CCNC(c2ccnc(C)n2)=O)CC2CC2)c1[N+](=O)[O-] C(C)(CO)(C(=O)NC(CC1CC1)CC1CC1)NC(CC(C)N(C)C)=O C#Cc1cccc(NC(=O)NC2CCCC2OCC)c1C#N C1(C(N(CCCCN(C(C(C)CC2CCC2)=O)C)C)=O)CC(C2CC2)C1 C(=O)(N1CC(O)CO1)c1c(NC(C2CC(C)(C)O2)=O)cccc1 c1(CC(N2CCC(O)(CNC(C(CC)SC)=O)CC2)=O)c[nH]c2ccc(F)cc12 C1(NC(CCOCCC)=O)CN(C(c2ccc(N(C)CC)cc2)=O)C2(CCC2)C1 N1(C(c2n(C=C)ncc2)=O)CCC(C(=O)N(OC)C2CCC2)C(C)(C)C1 C1(CNC(c2cc(CC)c(C)cc2)=O)CC12CCN(C(=O)C(C)(F)F)CC2 c1(CN2C(C)(C(=O)Oc3ccc(C(F)(F)F)cc3)CCC2)nnn2c1CCCC2 N1(C(C2(CNC(CC(CC=C)(C)C)=O)CCCO2)=O)CCc2nnnn2CC1 c1(C(=O)NC2CC(Cc3ccccc3)NC2=O)cc2n(n1)CCOC2 C(=O)(C(CNC(C12C(=O)C3CC1C2C3)=O)C(C)(C)C)N1CCC(OC)C(O)C1 Cc1cc(=NCC2CN(c3ccnn3C)C2)[nH]c(N2CC(C)CC(C)C2)n1 CN1CCC(C(=O)NC2CCCCC2C(N2CCCC(O)C2)=O)CC1=O N1(C(C)CC2(C)CC2)CCCC(C(=O)NC2CCCOC2)CC1 C1(N(C(=O)NCCOC)C)CC(=O)N(C2CC2C)C1=O Cc1[nH]c(C(C)(C)C)cc1C(=O)NC(C1CCN(C(C2CC3CC3C2)=O)C1)(C)C C=Cc1cncc(C(=O)NCC2COCCN2C(C2CC2C(=O)NCCO)=O)c1 Cc1cc(Cl)ccc1C(=O)N(C1CC(C#N)C1)CC(N1CC(c2cc(O)no2)C1)=O CC1CC(=O)NC1C(=O)Nc1cnn(CC(F)(F)F)c1C1CC1 c1(C(=O)NC(c2onc(-c3ccc(OC)cc3)n2)C(C)C)cc(C)ccc1CO c1(NCCSCC)ccc(-c2nc(C(C#N)C(C)(C)C)n(C3CCC3)n2)cc1 C=C1CC(C(=O)NCCC(=O)OC)(CNC(c2scnc2C)=O)C1 c1(NC(c2cccc(-c3n(C)ncn3)c2)=O)ncc(F)cc1C#N C1(C(N(CC(CC)(O)CC)C)=O)CC(C)(C)CCN1C(=O)C(C)NC(=O)NC C12(C(=O)NCc3c(OC)nsc3)CCC1CN(C(C1(NC(N)=O)CC1)=O)C2 N1(C(C2C(OCC)C2C)=O)CC(CO)C2(C1)CN(C(c1cnc3n1CCC3)=O)C2 c1(CC)ccoc1C(N1CCC(N(C(=O)CCCNC(=O)C2CC2)C)C1)=O NC1CCCC2(CC(C(N3CCN(c4nc(O)cs4)CC3)=O)C2)C1 c1(C(c2cccn2CC(C)C)NC(c2n(CC)nnn2)=O)ccc(OC)nc1 C=CCCCCCCC(=O)NC12COC(C1)C(NC(=O)C(F)CCC)C2 C1(CCC(=O)NCC2C(C(=O)OC)C2)CCCN(C(=O)CCn2ccnc2)C1 C1(n2cc(-c3cc(OC)ns3)nn2)CCC(C)(C)N(C(=O)CC(C2CC2)C2CC2)C1 Cc1cc(=NCCCCC(C)NC(C2CNC(=O)N2)=O)[nH]c(Cl)n1 N1(CC)CCCC1C(N1CC(COC)(NC(C2CCCSC2)=O)C1)=O C(=O)(CCCCCC#N)NC1C=CC(CC(=O)N(CC#C)CC2CCCO2)C1 c1(C(=O)NC(CCCNC(C=CCCC)=O)C)cc(C(N)=O)ccc1OC c1(CCC=CC(=O)NC(CNC(=O)CNC(N)=O)C2CCC2)ccccc1 CC#CC1CCN(C(C23CC(CO)(CN2C(C2CCCC(O)C2)=O)C3)=O)C1 CCCCC(CC)c1nnnn1C1COC1.c1(C(=O)N)cc(CC2CC2)on1 C1(N(C)C(c2cc(O)ncn2)=O)CN(C(C2CC3(CCO2)CC3)=O)CC12CC2 c1(OC)cccc(F)c1C(=O)NC1CCC1NC(=O)C(C)OCC(F)(F)F N1(C(Cn2cccc(N)c2=O)=O)CCC2CCN(C(c3ccncc3Cl)=O)C2C1 C1(N(S(=O)(=O)C2CCN(C(=O)OC(C)(C)C)C2)C(C)C)CCCCN(C)C1=O C12(NC(c3scc(C(=O)OC)c3)=O)CC1CN(C(=O)C(C(C)C)NC(C)=O)C2 C12(NC(c3cc(OC)n[nH]3)=O)CCCC1CN(C(c1n[nH]c(C)c1Cl)=O)C2 Nc1nccnc1C(=O)NC1CC1NC(=O)C(O)CC1CC1 CC1C(=O)Nc2ccccc2N1C(=O)C(=Cc1ccc2c(c1)OCO2)C#N c1(N2CCC(C)(C)S(=O)CC2)nc2c(c(=NC3CCc4nn[nH]c4C3)[nH]1)COC2 c1(CCC)ccc(C(N2CC(NC(=O)Cc3n[nH]c(C)n3)C3CC3C2)=O)c(O)n1 N1(C(C(CC)C(C)C)=O)C2CCC1CC(N(C(=O)C(C)n1cncn1)C)C2 C(=O)(C(F)CCC(CC)CC)NC(c1ccc(OC)cc1)CC(=O)OC N1(C(C2(CC)CCNC2=O)=O)CCN(C(c2cn(C)nc2Cl)=O)C(CO)C1 CC1(C)C(NC(=O)CCOC2CC2)CC1CNC(c1ccoc1Br)=O c1(C(=O)NCC(C)N(C(CC(=O)NCC#C)=O)CCC)nc(C)n(C)n1 c1(CC(=O)NCC(F)CNC(c2cn3c(n2)CCC3)=O)ccc(F)cc1F C#CCC(C)(CC)C(=O)N1CCC(C)(NC(=O)C=C2CCC(C)C2)CC1 CCCC(C)CCCC(=O)N1CC(OC)CC(NC(c2cscc2F)=O)C1 C(CCC1CCC1)(C(=O)N1CC(OCC2CC2)C1)NC(=O)Cc1cnoc1 c1(C(N(C2CCCN(C(CC(C(C)C)O)=O)C2)CCO)=O)nnn2c1CSCC2 C(C(C)(CNC(=O)Cc1ccc(-n2cnnc2)cc1)CO)OCC c1(NC(CCC2N(C(c3nn(CC)c(C)c3)=O)CCC2)=O)cc(C)cc(C)c1O N1(C(C2(N(C)C)CC2)=O)CC2C(CNC(=O)CC3C=CS(=O)(=O)C3)C2C1 C1(O)(C(C)N(C(C(C)(C2CC2)OC)=O)C2CC2)CCN(c2ncns2)C1 c1(N)cccc(N(C)C)c1.N1(CC)CCCC1C(=O)NCCC(C)NC(C(C)S)=O Clc1ccc(N2CCC(Cc3ccccc3)C2)nc1Br C1(COC)(CNC(=O)C(C(C)C)NC=O)CCN(C(C2CC3(CSC3)C2)=O)CC1 c1(C(N2C3(CNC(C(C(C)C)SC)=O)CCC2CC3)=O)cc2cc(Cl)ccc2[nH]1 c1(NC(CNC(C=C)=O)=O)cnc(C#N)c(Cl)c1.C12CC=CCC1C(=O)N2CC C1(NC(c2n(CC)ccn2)=O)CC12CCN(C(c1ccc(C)c(F)c1)=O)C2 CCC(C)(CC)C(=O)N1CC2CC2(n2cc(-c3cnn(C)c3COC)nn2)C1 c1(OC)c(C(=O)NC2CCCC2CNC(=O)C=Cc2cocn2)cc(Cl)cc1Cl c1(CCN(C)C(=O)NC2CC2CO)nc(C(F)(F)F)cs1 N1(C(C2CN(C(C(C)C)=O)C2)=O)CCC(NC(c2cccc(OC(C)C)c2)=O)CC1 c1(C(=O)NC(CC=C)CNC(=O)CCC2CCC(=O)NC2)cc(C)nc(C)n1 CCCCCCC(C)C(=O)NC(C(=O)NC(c1c[nH]ccc1=O)C)c1cccs1 N1(C(C2(F)CCCN(C(C(C)CC(F)F)=O)C2)=O)CCc2cnccc2C1 c1(CC(C(=O)NC(CC=C)(C)C)NC(=O)C(C)CC)cnn(C)c1O c1(OC)ccc2c(c1)CCCN2C(c1c(Cl)cccc1Cl)C(=O)NCC(C)C CCCC(C(=O)N(C1CCN(C(c2c(Br)n[nH]c2C)=O)CC1)CC)OCC C(C(O)CCNC(c1cc[nH]n1)=O)NC(C(C)n1cccn1)=O c1(C(N2C(CNC(CCC(C)SC)=O)CCC2)=O)ccnc2[nH]nnc12 c1(OC)ccccc1NC(C1CC(C)C1(C)C)=O C(=O)(C(C)CS(C)(=O)=O)NCC1(COC)N(C(c2ccn(CCC)n2)=O)CCC1 C1(NC(C2CN(C(=O)CN(C)C)CC(C)O2)=O)CC1C1CCCCC1 N1(C(C=Cc2cn(C)nc2)=O)CCCC(O)C1C(F)(F)F c1(N2CC(CNC(C3N(C(C)C)CCC3)=O)OCC2)ncc2ccsc2n1 C=CCCCCCCCC(=O)NCCCNC(c1cc(Cc2ccccc2)on1)=O C(=O)(C1CCc2c[nH]nc21)N1CCC(C=C)(C(=O)N(C)CCNC(=O)C(C)C)C1 CC1CCOC(C(=O)Nc2cccc(NC(=O)Cc3nc[nH]n3)c2)C1 c1(CC)nn[nH]c1C(=O)N(CCC(=O)NCC1CSC1)CCCO c1(C(=O)NC(CNC(COCC(C)(C)C)=O)C2CCC2)ccc2c(n1)COCC2 C(C(=O)NOC1CC1)(C(C)(C)C)NC(C(C)(C)CCF)=O.C1CC1 c1(CC)ccc(CN2CCC2COc2ccccc2C)cc1.C1(=O)CO1 C1(CC)CN(C)C(=O)CN1C(=O)C(CC(F)F)N(C(=O)Cn1nccc1C)C C1(NC(c2c(CC)[nH]cc2)=O)CC=C(C(=O)N2CCCCC(C)C2)C1 C1(C(=O)NC(CC=C)CC)CCN(C(C2OCCC2(C)C)=O)C1(C)C CCC(C#N)(CC)C(=O)NC(CNC(=O)CN1CCN(C)C(=O)C1)C(C)(C)C Cc1cc(C(=O)NCCN2CCC(NC(c3cnn[nH]3)=O)CC2)nc(C)c1 c1(NC(c2c(COC)ncs2)=O)cccc(CNC(=O)CC2CC2)c1 c1(C(N2CCC(NC(C3C(OC)(OC)CC3)=O)CC2)=O)c(C)oc(C)c1Br C1(CC(=O)OCC)CCCN1C(=O)CC1CCN(C(=O)Cc2cncnc2)C1 N=c1ccc(C(N2CCCCC2C(N2CCOC(CCO)C2)=O)=O)n[nH]1 C1(SC)CN(C(=O)C2=CCCS2)CC1NC(C1(C2CC2)CCC1)=O c1(-c2nc(-c3ccc(CC)cc3)nn2C2CCOC2)cccc2c1NC(=O)CC2 C1(NC(C(C)CC2CCCC2)=O)CN(C(=O)CO)CCC1C(F)(F)F C1(N(C(COCC)=O)CCO)CCN(C(c2ccnn2CC2CCC2)=O)C1 CC1=C(C(=O)N2CC(N(C(=O)C(n3cc(C)cn3)C)C)C3(CC3)C2)CCCC1 C1(CCC)(NC(c2csc(O)n2)=O)CCCN(C(=O)C(C)(C)c2ccccc2)C1 C1(C(N(CCCN(C)C)CCNC(C2(C)CCC2)=O)=O)CS(=O)(=O)CC12CCC2 C1(C(=O)NCC(C)OCC#C)CCN(C(C2COCCN2C)=O)CC1C N1(C(CC2C(CC)C2)=O)CCC(C2CC2)C1CNC(c1cnc(S)n1C1CC1)=O N1(c2nnc(-c3c(C)n(C)nc3)n2CC2CC2)CCOC2CCCCC12 CCC(C(=O)N1CCC(c2ocnc2Br)C1)Oc1ccccc1 C1(CCC)CCCN(C(C2CC23CC(NC(C2CCC2OCC)=O)C3)=O)CC1 C#Cc1ccccc1CC(N1CCCC(CC)C1C(=O)NCCCSC=C)=O CS(=O)(=O)c1csc(C(=O)NCC2CCC2NC(c2cncc(Cl)c2)=O)c1 CN1CCN(C)CC(C(N2CCC3(NC(C4(F)CCC4)=O)CCCC23)=O)C1 CC1OC2CCC1(C(=O)NCC1CCN(C(c3cncc(Cl)c3)=O)C1)C2 N1(C(C(CC=C)C)=O)CCN(C(C2CC(=O)N(CC)C2)=O)C(CO)C1 c1(C(=O)NC(COCC)C(=O)NCCS(=O)(=O)NC)coc2ccccc12 CCC(C(=O)NC1(c2ccccc2)CN(C(=O)CCCCCO)C1)C(C)C CC1(C)CN(C(C2CCC(C(N)=O)O2)=O)CC1NC(=O)CC12COC(CF)(C1)C2 c1(C(=O)NC2CCCC(NC(CC3ON=C(C)C3)=O)C2)cc2ccsc2s1 N1(C(C(C)NC(C)=O)=O)CCCC(C)(C)C1C(=O)N(C)CCc1cc[nH]n1 C1(C(C)NCC(O)COc2ccc(Cl)cc2Cl)CC2(CCC(F)(F)CC2)C1 N1(C(COC(C)=O)=O)CCC2(CC1)CCN2C(c1ncccc1Br)=O CC1(C)CCC(CNC(=O)Cn2cccn2)N(C(=O)Cn2cc(F)ccc2=O)C1 N1CCOCC1CC=O.C(C(=O)NOCC(O)C(C)C)C1CC(C)C1 Cc1nc(C)c(C(=O)NCC=C2CCN(C(=O)CC(F)(F)Cl)CC2)[nH]1 c1(N2CCCC(CNC(c3cccc(CC)n3)=O)C2)cc(C)nc(C(C)(C)C)n1 C1(NC(C2(CNC(c3cc(C)ns3)=O)CC=CC2)=O)COC2(CCC2)C1 C1(C(=O)NC(CC)CN(C)C(c2cnn(CC(F)F)c2)=O)CCCC(=O)O1 N1(Cc2ccc(N(C)C)nc2)CCC(F)(F)C(NC(c2ccccc2)=O)C1 C1(NC(c2ccc(C#C)cc2OC)=O)CCN(C(=O)CC(C)OC)CCC1(F)F C=CC(C)(CC)C(=O)NCCC1CCN(C(c2cnc(C(C)=O)s2)=O)C1 c1(C(=O)NC(C2(O)CN(C(=O)Cn3cc(C(F)F)cn3)C2)C)cc(C2CC2)cs1 N1(C(CNC(C2C(C)C2)=O)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 CCCC(C(=O)NC(C1(C)CCN(C(c2cncs2)=O)C1)C)c1cccc(Cl)c1 C(=O)(C1=NOC2COCC12)NC1C(NC(c2c(C)nccn2)=O)CCC1 C1(NC(c2cnc(OC)c(Cl)c2)=O)CCCC12CN(C(c1ncc(F)cn1)=O)C2 c1(C(=O)OCC)ccc(C(=O)NCCCC(C)NC(C2CCOCC2)=O)cc1 N#Cc1ccc(NCC(N2CC=CC2C(N2CC3CC2(C(F)F)C3)=O)=O)cc1 C1(C(=O)NCC2C(C)OCC2)CC12CCN(C(c1cccn1C)=O)C2 N1(C(=O)OC)CCC(NC(C2CCCN(C(=O)CNC(=O)C(C)CO)C2)=O)CC1 C1(C(N(C)CC2CN(C(C3(S(N)(=O)=O)CC3)=O)CCO2)=O)CCCCCCC1 C(C(F)(F)C(=O)NCC(CCOC)NC(c1cnc(O)n1C)=O)OC C(C(=O)NCC(C1CCC1)NC(c1ccc(C(C)=O)[nH]1)=O)(C(C)C)SCC Cc1cc2sc(C(N3CCCC3CCNC(c3cncs3)=O)=O)cc2s1 c1(NCCn2cncn2)nccc(=NCCCC2CCC3CC23)[nH]1 c1(C(C(=O)NCC(=C)C)N(C2CCCC2(C)C)C)ccc(Br)nc1 c1(CC(=O)N)cccn(C2CC2)c1=O.C1(CN(C2CCCC2)CCNC)CN(C)C1 N1(C(C2N(C(CNC(=O)C3CC3)=O)CC(O)C2)=O)CC2CC=CCC2C1 CC(C)(O)C(F)C(=O)N1CCC(CCNC(=O)CCC2CCCO2)C1 c1(C(=O)N)cc(N)ccc1O.N1(C(CCC2CC(NC)C2)=O)CCC(n2cccn2)C1 c1(C(N2CCCC(CNC(CC3N(C)CC=CC3)=O)C2)=O)ccn2nnnc2c1 N12CCN(CC1)C(C(F)(F)F)CNC(C)(C1CC1)C2=O.S(C)(=O)(=O)N.C(C)(=O)OC C(=O)(C(C)(C)CC(F)(F)F)N(CCC(C(C)C)NC(c1cc(C)cc(O)c1)=O)C C(c1cnc(O)nc1O)=CC(=O)OCNC1CCCC(C(C)(C)C)C1 c1(CN(C(=O)C(O)CNC(=O)CCOCCN(C)C)C)cc(=O)cc[nH]1 C(CC(C)(C)C)(C(=O)NCC1(C)CCCN(C(C2(n3ccnn3)CC2)=O)C1)OC Cc1ccc(OCC(O)CN2CCC(C)(CNC(c3cc(C)sn3)=O)C2)cc1 C(=O)(C(C(C)(C)C)c1cc(F)cc(F)c1)NC1(CCNC(C(CC)OC)=O)CC1 C(c1ccccc1)=C(C(=O)N(CCCOCCNC(CCC=C)=O)C)OC C1(C(=O)NCCOCCN(C(C2(COC)COC2)=O)C)CCC(C(F)(F)F)CC1 C12(NC(C(C)Cn3ccnc3)=O)CCOCC1CN(C(c1csc(=N)[nH]1)=O)C2 C1(NC(=O)Cn2nc(C(F)F)cc2C(F)F)CCN(C(=O)C2COCCO2)O1 Cc1cc(Br)cc2nc(CN=c3[nH]c(N(C)CCc4cccs4)nc(=N)[nH]3)[nH]c12 C1(O)(C(C)NC(CC(=O)NCC#C)=O)CCN(C(c2nc(C)nn2C)=O)C1.C1(C)CC1 c1(C(=O)NCC(C)(CC(C)C)NC(C=CCCC)=O)c(C)ccc(C)c1N C(CCN(C)C(C1CCCC1OC)=O)(C(C)C)NC(c1cc(C(CC)C)no1)=O N1(C(CCc2cc(C)no2)=O)CCC2(CCN(C(c3c[nH]c(C(F)F)n3)=O)C2)C1 C(=O)(C(CNC(=O)CC1CC(C(F)F)C1)c1ccccc1)OCC C(C(=O)N1CCC(C(C(C)C)NC(c2ccc(=N)[nH]c2)=O)CC1)(C(C)C)SCC c1(CC(=O)NC2CCCC2CNC(C2CCCC3CC23)=O)ccc(O)c(F)c1 c1(C(=O)NCCN(C(=O)CSC)CCC)cc(Br)n2ccccc12 c1(NC(c2ccc(-c3ccc(NC(C)=O)cc3)nc2)=O)ccc(F)nc1F c1(OC)nc(C)ccc1C(N1CCCC(C(=O)NCCC#N)CC1)=O c1(C(=O)NCC(C)(C)OCC(=O)NC(CC)(C)C)ccc(C)cn1 Cc1c(C(N2CC3(CC(NC(C4CC4Cl)=O)C3)C2)=O)oc2cc(Cl)ccc12 C1(NC(C(c2ccccc2)=C(C)C)=O)CC2CCC(C1)N2C(C12CCCC1C2)=O c1(OCC)ccc(OCC(=O)N(C(C)CNC(=O)C(F)n2ccnc2)C)cc1 c1(C2C(CNCC(C)C)CCC2)cccc(Cl)c1 O=C(CCCCC(F)F)NC1CC2CCC1CN(C(c1cnsn1)=O)C2 c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2F)cc(C)c(Cl)c(C)c1 c1(OC)ccc(Cl)c(C(c2noc(-c3cc(C(N)=O)cs3)n2)C)c1 N1(C(CCc2cnc(C)s2)=O)CCC(C2CC(NC(c3nc(Cl)cs3)=O)C2)C1 N1(C(C)=O)CCCC1C1CCCN1C(N1CCC2CCCC2C1)=O c1(CCC(=O)NCC2CN(C(Cc3cnc(C)o3)=O)C(C)C2)cccc(C#N)c1 N1(C(c2nc[nH]c2C(F)(F)F)=O)CCC2CCC(C1)N2C(C1(CO)CC1(F)F)=O c1(Cc2cn(CC(=O)NC(CCNS(CC)(=O)=O)(C)C)nn2)cccc(C(F)F)c1 C(CN=c1[nH]c2c(c(=NC(C)c3ccc(N(C)C)nc3)[nH]1)COC2)SCC C1(C(N)=O)CCC(C(=O)NCCC2CCC(NC(=O)C=CCn3cncn3)C2)CC1 Cc1cc(CN2CCCCC2CNC(=O)CCc2cnc[nH]2)ccc1F CC(CC(=O)N1CCC(F)C(NC(c2ccc3c(c2)OCO3)=O)C1)C(F)(F)F C(CC(F)(F)C(=O)NCC1CCC2(CCC2)C1)n1cc(CCNC(N)=O)nn1 c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2)cc2ccc(Cl)cc2s1 c1(CNC(C(C)CO)=O)nn(C)c2c1CN(C(=O)Cc1ccccc1Br)CC2 c1(C(=O)NCC(CNC(C(Cc2ncn(C)c2)O)=O)(C)C)cc2scc(Cl)c2[nH]1 C(=O)(C(C)C(C)(C)C)NCCC(C)(C)NC(C(c1cccnc1)C)=O n1(CC)nc(C(=O)NC(C2CC=CCC2)C(=O)NCCc2cc(C)ns2)cc1C c1(C(=O)NC2CC(NC(C(C3CCOCC3)C)=O)C2)cc(N)c2ccccc2n1 c1(C(=O)NC2CN(C(Cc3ccc(OC)cc3)=O)CC2C)ccc(Br)cc1F C1(O)(C(=O)NC(C)CCCNC(=O)CCC2CC2(F)F)CCCCC1 Cc1cc(Br)ccc1S(=O)(=O)N1CCC(C(=O)Nc2c(C)cccc2[N+](=O)[O-])C1 c1(C(=O)NCC2C(NC(C(F)=C(C)C)=O)C2)ccn(CC(F)F)c(=O)c1 c1(-c2cn(C)nc2)ccc(CNC2CC3CCC2C3)cc1 c1(C(C)Nc2ncnc(NCc3c(C)nco3)c2C)ccc2c(c1)CCCO2 O=C(C1=CC2CCCC12)NC1CCCCC1NC(c1ccc(CO)nc1)=O C1(NC(=O)CC(F)F)CCCOC1C1CCN(C(c2ccoc2Cl)=O)CC1 N1(C(Cc2cc(CC)no2)=O)CC(NC(=O)CN2CCC(C)CC2)C2(CCC2)C1 c1(CCC(=O)NCC(CC)NC(c2ccn(C)c(=O)c2)=O)c(O)nc(=N)[nH]c1C c1(CCC(=O)NC2CCC(N(C(COCC#C)=O)C)C2)ccnc(Cl)c1 CCC(CNC(c1[nH]cc2c1CCC2)=O)N=c1ncnc(NC(C)=O)[nH]1 C1(CNC(c2ccc(COC)[nH]2)=O)C(C)CCN1C(C1CC1C(C)C)=O N1(C(C2ON=C(C)C2)=O)CCC(C(=O)NCc2[nH]nnc2C)C12CC2 c1(C(N2C(C(=O)NC(CC)C(C)O)CC(C)C2)=O)c(C)cc(OC)cc1C c1(C(=O)NCCCC2N(C(CC(=C)C)=O)CCC2)cc(Br)ccc1OC c1(C(N2CCC(C(N3CC(C)NC(=O)C3)=O)C2)=O)cccc2nc[nH]c12 N1(c2cc(C)nc(Cl)n2)CCS(=O)(=O)C(CCNC(=O)CN2CCCCCC2)C1 c12ccccc1OC(=O)CC2.c1(CN(C)C)ccn(-c2ccccc2)n1 c1(OC)cc(C#N)cc(Cl)c1OC(=O)C(O)CC[S+](C)C N1(C(CCCC2C(C)C2)=O)CCCC(CCC(=O)NCc2ccoc2C(C)C)C1 C1(NC(=O)OC(C)(C)C)CCCN(c2nccc(-c3cccc(Br)c3)n2)C1 Cc1cccn(CC(=O)NC(C2(CNC(C3CCOC3(C)C)=O)CC2)C)c1=O CC(C)C(C#N)C(=O)N1CCC(NC(C2CCC(C)CC2)=O)C1 c1(C(N2CCCC(NC(c3n(CC)ncc3Cl)=O)C2)=O)cc(S(N)(=O)=O)c(C)o1 c1(NC(CN2CCCC(OCc3n(C)ccn3)C2)=O)c(F)ccc(N)c1F c1(C(=O)NCC(F)CNC(C2(F)CC2)=O)nc[nH]c2ncnc1-2 C1(CNC(CCc2n(C)ncc2)=O)CC(C)(C)CN1C(=O)CC1(CO)CC1 N1(C(=O)CC2CCCCC2I)CC(CO)Cn2ccnc21 c1(CN2C(C(=O)Nc3nc(OC)cnc3Cl)CC(=C)C2)cccc2ccoc12 C1(NC(=O)Cn2cnnn2)CC2CC1CN(C(=O)Cc1ccc3c(c1)CC3)C2 C(=O)(C1=CCCCO1)NCC1(F)CN(C(c2c(C(=O)OC)cccc2)=O)C1 CCC(C(=O)N1CC(CCCCOCc2cc(C)no2)C1)OC.C1(=O)CN1CC C1(NC(c2cnn(C)c2Br)=O)CC2(C1)CC(N)C2 CC(C)CCCC(C)C(=O)N1CCN1C c1(NC(C2N(C(=O)Nc3ccc(C)cc3)CC(O)C2)=O)cnc(Cl)c(Br)c1 c1(CC)nc(N2CCC(NC(c3c[nH]cc(Cl)c3=O)=O)C(C)C2)cc(C#N)n1 C#CCCCC(C)C(=O)NCC(C)(C(C)C)NC(=O)C(=O)NCC(F)(F)F C(CCCC(CO)NC(=O)CCOCC1CC1)NC(c1onc(CC)c1C)=O C1(CC)C(C(=O)NCC(C)(C)C2CC2)CCCN1C(=O)CC1CCOC1C c1(C(N2CCC(C(C)NC(C(C=CC)O)=O)CC2)=O)c(F)cc(OC)c(F)c1F c1(N2CC(NC(C(C)Oc3ccc(C)cc3)=O)C(C)CC2)ncc(C#N)cc1Cl Cc1ccn2c(C(=O)N(C)C(c3cn(CC4CCCC4(F)F)nn3)C)cnc2c1 C(=O)(C(F)C(C)(C)O)NCC(CCOC)NC(=O)C(C)(C)C(C)C CC1(C)CN(C(N2CC3CCC2CC3Br)=O)CC(CO)O1 CN=S(C)(=O)CCNS(N(C)CCO)(=O)=O.C1(=O)CN1C(C)CN(CC)CC C1(C)(CC(N2CCC(CNC(C(CCOC)C)=O)CC2)=O)CCCCCC1 c1(C(=O)NCC2N(C(CN(CC)CC)=O)CCCC2)cc2ccc(F)cc2o1 C12(C(N3CC(NC(CCOCCC)=O)(COC)C3)=O)CC(=O)N1CCS2 C1(C(=O)NC2(C(C)C)CC2)CC(NC(C2(n3cccc3)CC2)=O)CCO1 n1(CC)ccc(C(N2CCCC2CCC(=O)NC2CC3CC3C2)=O)c1C N1(C(C(C)CC2CC2)=O)CC(F)CC1C(=O)NCCS(C)(=N)=O c1(OC)c(Br)ccc(C(c2nnnn2-c2ccccc2)NCC2(CF)CC2)c1F N(C1CCc2cccc(Br)c21)C(=O)NCc1c(C(C)(F)F)cccc1 N1(C(c2c(C)csc2)=O)CC2(C1)OC1(C)CC2(NC(=O)C(C(C)C)NC=O)C1 C1(OC)CN(C(=O)CSC(C)C)CC1NC(=O)CC(c1ccc(C2CC2)cc1)C C1(C(N(C)CCOCCCNC(C2(C)CC2C(F)(F)F)=O)=O)CNC(=O)N1 N1(C(C2CCS(=O)(=O)N2)=O)CCC=C(CNC(C2(Cl)CCC2)=O)C1 C1(NC(=O)C=C2CCOCC2)CCSC12CN(C(c1cccc(C(F)F)c1)=O)C2 N1(C(C2CC(O)C23CCOCC3)=O)CC(S(=O)(=O)CC(F)(F)F)C1 O=C(CC(C(F)(F)F)c1ccc(F)cc1F)NC1CC1c1ccc(F)cc1 C1(NC(C2(F)CCOC2C)=O)C2CCN(C(c3cc(COC)ccn3)=O)CC12.C(=O)C1CC1 c1(C(N2CCC(C(C#C)C)CC2)=O)ccc2c(c1)OCC(F)(F)C(F)(F)CO2 c1(C(=O)NC(C(C)NC(CSC)=O)(C)C)ccnc(N2CCCC(C)C2)c1 C=CC1(C(=O)NC2CC(C(C)(C)C)C2)CCN(C(C2C(C#N)C2(C)C)=O)CC1 C1(C(=O)OC)CC2CCC1CC2NC(=O)NC1(CC(=O)OC(C)(C)C)COC1 c1(OC)cc(Cl)cc2[nH]c(C(=O)N(C(C)CNC(C3CCCO3)=O)C)cc12 CC1CCN(C(=O)C(=O)NC2C=CCN(C(c3ccc(C#N)[nH]3)=O)C2)CC1 N1(C(CNC(=O)OC)=O)CCC(CC(C)NC(C2(CO)COC2)=O)CC1 N1(C(CCCCCCCC)=O)CCC2OCCN(C(C3CCCCN3C)=O)C2C1 C1(C(N2CC(O)(CNC(c3n(C)nnc3)=O)C2)=O)CCc2n[nH]cc2C1 Cc1cc(-c2nn[nH]n2)ccc1C(=O)NC1CN(C(c2ccccc2)=O)CC1O C1(N(C2CCNCCC2C)C(c2c(COC)onc2)=O)CCc2n[nH]cc2C1 Cc1ccc(C)c(CCCC(=O)NCCC(O)CNC(C2(C)CC2(F)F)=O)c1 c1(C(=O)NC2CCC(NC(C3CC(C(=O)OC)C3)=O)CC2)cc(F)cc(F)c1 C(=O)(CCC(=O)c1ccc(O)cc1)NCC(CN(C(=O)C1=CCCO1)C)O N#Cc1ccc(N2CCCC(C(=O)NCCc3cnc(S)nc3)C2)cc1 C1(CNC(C(C(COC)C)C)=O)CN(C(=O)CCCCC#N)CCC12CCC2 n1(CC(=O)NC(CC=C)CNC(=O)C=Cc2cn[nH]c2)cnc2c1CCCC2 N1(Cc2c(C)nc(CC)o2)CCC2C(CCCN2C(=O)CCc2cnn[nH]2)C1 C1(NC(CCCOCC)=O)COCCC1C(=O)NC1C=CCCC1 C(=O)(N=c1[nH][nH]c(C)c1C)C1C(NC(=O)NC(Cc2cccc(OCC)c2)=O)C1 N1(CCCSC)C(=O)CN(CCCCn2cncn2)C1=O C=CC1(NC(=O)CCN(C(=O)C(=O)NC(C)C)C(C)C)CCOCC1 c1(C(C)CC(=O)NCC(C)N(C)C(C2CCSCC2)=O)ccccc1F c1(C(=O)NC(C2CCCN2C(=O)CCc2cc(Cl)no2)(C)C)coc2c1COC2 c1(C(=O)NC2CC(C)N(C(=O)Cc3ccccc3Cl)CC2)nccn2ccnc12 C1(NC(CC(COC)C)=O)(CNC(=O)C(C)OC)CC2CCC1CC2 CC1(C)CN(C(C23CCC(CC2O)C3)=O)CC1CNC(c1n[nH]cc1Cl)=O CC(=O)CCCC(C)C(=O)NC(CC(=O)NCCc1cnco1)C(F)F CCC(C)CC(C(=O)NC1(C)CN2CCC1CC2)NC(=O)CCCC(C)C N1(C(=O)CC2CCCCCC2)CCN(C(c2cc(Br)cnc2O)=O)C(CF)C1 Clc1ccnc(NCC2CC3(CCOC3)C2)c1I c1(C(=O)NC2CN(C(CCc3nnc(C)n3C)=O)C(C)C2)cccc2nc[nH]c12 c1(C2COCC(C)O2)ccc(C2(NC(c3cncc(C#N)c3)=O)CC2)c(F)c1 N1(CCCC(=O)NC2CCC2NC(=O)CCC2CC(F)(F)C2)C(=O)CNC1=O N1(C(c2ccc(Cl)o2)C(=O)NC2CCOC2)CC2CCC1C(O)C2 C1(CC(=O)NC2CCN(C(c3ccc(F)o3)=O)CC2F)CCCC2(CCC2)O1 c1(C(N2CC(NC(=O)C(F)(F)c3ccccc3)C(O)C2)=O)cc(F)ccc1Br c1(C(N2CCCC(C(C)(C)O)C2)=O)ccc2c(n1)CN(C(=O)C1CC1)CC2 C1(O)(CN(C(COCC(C)C)=O)C)CN(C(C2CCN2S(C)(=O)=O)=O)C1 C#CC1CCCN1C(=O)NCC1COCC1c1ccc(Cl)cn1 c1(C(=O)NCCC2(O)CN(C(COCC#C)=O)C2)cc(F)cc(Br)c1 c1(C(N2CCN(C(C3N(CCC)CCC3)=O)C(CC)C2)=O)cc(C#N)c(C)cn1 CCC(C)C(C)C(=O)N1CCC(CNC(c2cc(C3CCCC3)[nH]n2)=O)C1(C)C C1(CC(=O)N(C2C(C)CC2)Cc2ccccc2)CNC(C)(C)CO1 c1(OC)cnc(C(=O)NC2CCN(C(=O)C3=CSCS3)CC2)nc1 Cc1c(C(=O)NC2CC3CCC(C2)N3C(=O)C(C)C)oc2ccc(Br)cc12 N1(C(COCCCC(C)C)=O)CC(NC(=O)CC2(C)CCCCC2)C(F)(F)C1 N1(C(C2OCC(C)(C)C2)=O)C2CCC1CC(C(=O)NCCCc1nncs1)C2 c1(C(=O)NCC2C(NC(c3cc(Br)co3)=O)CC2)cccc2[nH]ncc12 N1(C(C=C(CCC)C)=O)CCCC1CC(=O)N(CC(C)(C)C)C1CC1 C1(CC)CN(C(=O)NCC2CCCN2C)CC1CO c1(C(=O)NC2C(C(N(C(C)C(=O)NC)CC)=O)CCOC2)cccc(C)c1O c1(C(=O)NC(C)CC(C)NC(C2CCS2(=O)=O)=O)ccc(-n2cccn2)c(F)c1 N1(C(C2(C(=O)O)CCOC2)=O)CCC(C2(O)CCOCC2)CC1 c1(CNC(=O)CCc2ccccn2)cccc(C(=O)NC2(C(=O)O)CCC2)c1 N1(C(C(CCC)OC)=O)CC(NC(C2CCC3(CCC3)CC2)=O)C2CCCCC12 c1(-n2cc(CN(C(=O)Cc3ccnc(Br)c3)C)nn2)ccc([N+](=O)[O-])cc1 C(=O)(C=CC(C)NC(C1CSC1)=O)N(C)CC C1(C(=O)NCC(=C)Br)(CC)CCN(C(c2cc(C)nc(O)n2)=O)CC1 N1(C(=O)Cn2ccc(C(F)F)n2)CCN(C(C2CCCC(F)C2)=O)C(CO)C1 c1(C(=O)NC(CNC(C(C=C)(C)CC)=O)(C)CC)ncc(C#N)cc1C Cn1ncc(C(N2CCCCC2CCNC(c2ccc(Cl)nc2)=O)=O)c1C1CC1 N1(C(c2c(O)ccc(C)c2)=O)CCC2CN(C(c3cc(Cl)no3)=O)CCC12 CC1(C)CN(C(=O)CN2C(=O)CCC2=O)CCN(C(=O)C#CC2CCCCO2)C1 Cc1nc(C)c(C(=O)N(C2CCCN(C(C3(C(C)C)CC3)=O)C2)CCF)[nH]1 CC(C)C(F)(CNC(c1cc(F)cnc1O)=O)C(=O)NCc1cncc(O)c1 c1(NC2C(c3n(C)nnn3)CC2)cccc(-c2ccon2)c1 CC(C)(C)CCCCC(=O)NC1CCC(NC(=O)CC2CC(=O)C2)CC1 CCC(CC(F)F)C(=O)NC(C1(C)CC2(CCC2)C1)C(=O)O Cc1nc2c(C(=O)NC3CC3CNC(C3CCCCC3O)=O)ccnc2[nH]1 C(c1cn(C)c(=O)n(C)c1=O)=CC(=O)NC1CN(C(CC(C(=O)OCC)C)=O)C1 c1(C(=O)CO)ccc(C(F)(F)F)nc1.C1(N(CCO)C=O)CCCN(CC(F)(F)F)C1 c1(C(=O)NCC(CC)NC(C2CCCN2C(C)C)=O)cccc2occc12 CC(C)C(C(=O)N(CCCNC(=O)CC1(C)CC1)C)NC(=O)Cc1ccccc1 c1(C(=O)OC)ccc(N2CCC(C(N)=O)C2)nc1Br C=CCC(C(=O)NCC=CC(=O)N(C(C)CO)C)NC(C)=O c1(-c2cn(CC(N3C(C(=O)OC)(CC4CC4)CCC3)=O)nn2)ncc(F)cc1F CCC(CC)(C(=O)N1CCC(C)(CCNC(=O)C=Cc2ccccn2)C1)C(C)C Cc1cc(Cl)c(C(=O)NC(C2CCOC2)CNC(c2cnc(S)[nH]2)=O)cn1 C(=O)(CC1CCOc2ccccc21)N1CCN(C(c2c(CC)con2)=O)C2C1C2 C=CC(C)(C)C(=O)NC(CNC(=O)C(c1cnccc1C)(C)C)CC N1(C(CCCCC(=O)NC)=O)CCC(NC(=O)C=Cc2cnc[nH]2)C2(CCC2)C1 C(CC(C)(C)C(=O)N1CCC1C1CCC1)NC(C(SC)SC)=O Cn1cnn(CCC(=O)NCC2COCCN2C(=O)C2=NOCC2)c1=O Cc1cccc2c1CN(C(=O)C(c1ccoc1)NC(=O)CC#N)C2 c1(CC)ccc(C(=O)NC23COC(C2)C(NC(=O)C(C(C)C)SC)C3)cc1Cl c1(-n2cc(CCCNC(c3cc(Cl)sc3Cl)=O)nn2)ncc(Cl)cn1 C1(N(C)C(C2CCC3CC3CC2)=O)CCCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 CCC(C(c1nnnn1C)NCC1(NC)CCCC2CC12)C(C)C c1(C(N(CCC(=O)NCC(=O)NC(C)C)C2CC2)=O)sccc1C#N C1(OC)CC(NC(c2cccc(F)c2)=O)CN(C(=O)CN2CCCC2)C1 Cc1noc(C)c1CC(=O)NC1CCC1NC(=O)CC(C)(F)F C1(CN(C(c2c(OC)c[nH]n2)=O)C2CC2)CCCCN1C(=O)CCNC(C)=O c1(SCCC(=O)NCc2cccnc2Cl)ccccc1C(=O)NC1CC(CC)C1 C1(NC(COCC)=O)CC12CCN(C(=O)CCC1CC(C)(C)CO1)CC2 c1(C(N2CC(C)(NC(c3cccc(OC)c3F)=O)C2)=O)cc(S(N)(=O)=O)co1 C(C(C)(C)CC(=O)NC1CCOC1C)NC(C=Cc1ccc(C)o1)=O C1(CNCc2c(C)ccs2)CC2CC2N1C(=O)CCCC1CCN1 C1(C(=O)NCC2(OCC)CC2)CN(C(=O)CC2CCCCO2)CC(C)O1 c1(CC(N2C(CNC(CC(C)CN(C)C)=O)CCCC2)=O)cc2ccccc2s1 C1(Br)(C(=O)OC)CC1C(=O)NC1CC1NC(c1ccsc1)=O c1(CC(=O)NC(CNC(c2[nH]c(CC)c(Cl)n2)=O)(C)CO)cn2c(C)cncc2n1 CCCC(CC)C(=O)NCC1(F)CC(NC(=O)C(C)(C)N2CCCC2)C1 Cc1cc(C)c(CNC(N2CCOCC2c2cn[nH]c2)=O)s1 c1(OC)ccc2c(c1)CCC2C(=O)N1CCC(CNC(=O)C2=CCC2)C12CC2 c1(C(=O)NCCCCNC(c2nnc(OC)s2)=O)c(C)coc1-c1ccccc1 CC(C)C(CCN(C(=O)COCC1CC1)C)NC(c1ccc(-c2cccs2)s1)=O c1(C(=O)NCCN(C(=O)Cc2ccnn2C2CCC2)C(C)C)ccc(Cl)c(N)c1 C1(C(=O)NC(c2c(C)cccc2Br)C)C(C2CC2)CCN1C(=O)CC1(N(C)C)CC1 CCC(CC(=O)NCC1CC(C)CN(C(=O)Cc2cnn(C3CC3)c2)C1)C(F)F n1(CC(=O)OC)cnc(C)c1C(=O)NC1CCOCC1NC(=O)C(C)CSC C(C(C)CN=c1cc(Cl)nc(CC)[nH]1)NC(C(CCCC)(C)F)=O c1(C(=O)OC)cn2c(n1)CN(C(c1ccnc(OC)c1F)C(=O)NC1CC1)CC2 C1(C(=O)NCCC(C)NC(c2cc(C3CC3)ncn2)=O)(COC)CCC(=O)N1 C(C(CNC(=O)C(C)OC(C)(C)C)S(C)(=O)=O)NC(c1ccc(C)n1C)=O CC(C)CC(CN(C)C)CC(=O)NCCNc1ccccc1F C1(NC(c2ccc(C(CC)C)cc2)=O)(CO)CCCN(C(=O)CC(=O)OC)C1 C(CN=c1[nH]c2ccccc2s1)CCNC(CCN1CCCC(C(N)=O)C1)=O C1(n2cc(C(C)N(C)C(c3cc(C(F)F)no3)=O)nn2)CCCCCC1 N1(C(C2C(CNC(C(C)=CCC)=O)CC2)=O)CC2(CCN(C)CC2)C1 N1(C(C(CC=C)(C)C)=O)CCC2(COCCN2C(=O)C(C)n2cccc2)C1 N1(C(C(CO)NC(N)=O)=O)CCC(=CCNC(C2CC23CCOC3)=O)CC1 CC1(C)CC(NC(c2cc(C(F)F)[nH]n2)=O)CN1C(=O)CCOC1CC1 Cc1cc(S(=O)(=O)NCCCNc2cccnc2)c(C(=O)O)cc1Cl Cc1csc(Cl)c1C(=O)NCC1(C(C)(C)C)CCN(C(C2(CF)CC2)=O)C1 C1(CNC(C2N(C(C)=O)CCC2)=O)CC2CCC1N2C(=O)CCC(F)F N1(C(CCSCCC)=O)CCC=CC1C(=O)N(CC(O)CC)CC N1(C(C(CCC)OCC)=O)CC2COCC2(C(=O)NC(C)CCC(F)(F)F)C1 Cn1ncc2c1CC(C(=O)NCC1COCCN1C(C13CC(C)(CO1)C3)=O)CC2 C(CCC(N)=O)(C(=O)NC1CCN(C(c2coc(C#N)c2)=O)C1)N(C)C Cc1ncccc1C(=O)N(C1CC(NC(c2c(CO)noc2C)=O)C1)C CC(C)(C#CC(=O)N1CC2CSCC2C1)CNC(C1(C)CC=CCC1)=O Cc1ccc2c(c1)C(NC(C1CC1F)=O)CCCN2C(c1ncco1)=O CC1NC(=O)CCC1NC(C1CC(O)(CN(C(C2CCO2)=O)C2CC2)C1)=O c1(C(=O)NCCN(CCCCCC)C(=O)C(C)C2CC2)c[nH]c2cccc(C)c12 c1(CC(=O)NCC(O)CCNC(c2cc(O)ncn2)=O)ccccc1Cl C1(c2n(CC(=O)OC)nnn2)(Nc2ccc(Br)c(C)c2C)Cc2ccccc2C1 C1(C(=O)NCC2N(CC)CCC2)CN(C(c2nnc(S)n2C)=O)CC1C c1ncnc2cc(I)sc12.N1(C(C)=O)CCN(c2ncc3ccsc3n2)CC1C#N C#Cc1ccc(C(=O)NCCN(C(=O)C(c2ccc(C)s2)C)C(C)C)c(F)c1Cl N1(C(C(C=C)(F)F)=O)CCN(C(c2cccn2CC)=O)C(CCCC)C1 NS(=O)(=O)c1ccc(C(=O)Nc2ccc(I)c(F)c2F)nc1 Cc1cc(NC(c2ncoc2CNC(=O)C(C)(F)F)=O)cc(F)c1 C(c1cccc(O)c1)=CC(=O)N(C)CCN(C)C(c1cncc(C(F)F)c1)=O Cn1c(O)ncc(C(N2CCCCC(CNC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)c1=O C(=O)(C(C)(C)S(=O)(=O)C1CC1)N(C1CN(C(C2(CCCC)CC2)=O)CC1F)C CCC(C(=O)N1CC(C(C)(C)O)(CNC(=O)C(F)n2ccnc2)C1)NC(C)=O c1(C(=O)NCCC2(N(C(=O)CN3CC4CC4C3)C(C)C)CC2)cc2c(Cl)nccc2o1 Cc1cc(C#N)nc(N)c1C(N1CC2(c3ccccc3)CCC1C2)=O C(=O)(N1CCCc2nncn21)C1CCN(C(Cc2cnc(C)s2)=O)CC1(C)C C(C)(C(C)C(=O)NCCCS(C)(=O)=O)NC(C1CC(O)(CC#C)C1)=O c1(C(C)NC(C(C2N(C(C(C3CC3)OCC)=O)CCC2)(C)C)=O)ccc(C)cn1 c1(C(=O)NC2C(C)(C)CN(C(=O)C(O)P(C)(C)=O)C2)coc2ccccc12 Cc1ccc(C(N2CCCC2(C)CNC(C2CCCC23CC3)=O)=O)nn1 Cc1cc2sc(C(=O)NC(C3CCCN3C(C3CC34CCCC4)=O)(C)C)cc2s1 c1(-n2c(C(n3nccn3)C)nc(CC)n2)ccc2c(c1)CCO2 c1(C(=O)NCCC(C)NC(=O)Cc2nnc(O)s2)cccc2nccnc12 N1(C(C)=O)CCOC(C)(CNC(=O)C(c2cccc(C)n2)(F)F)C1 c1(NCC(C)NC(c2c(C)sc(C(F)(F)F)n2)=O)nc(C(C)C)nc2[nH]ccc12 C=CC1(C(N2CCC(N(C(C3CC4(C3)CC(O)C4)=O)CC)C2)=O)CCCCC1 N1(C(C=C(COC)C)=O)CC2CCC(CNC(=O)COc3ccsc3Cl)(C2)C1 C1(SC)CCCC(F)(F)C1.c12nc(ns1)C(=O)NCCN2CCOC Cn1cc([N+](=O)[O-])cc1C(N1C2CCC1CC(CCNC(=O)C1=NOCC1)C2)=O c1(-c2nc(C)sc2)cc(C(=O)NCC2CC2NC(=O)CC(C)(F)F)c(C)o1 Cc1nn2ccccc2c1C(=O)NC(c1cn(-c2ccc(F)cc2)nn1)C c1(OC)ccc2c(C)c(C(=O)NC(C3(O)CCCCC3)C)oc2c1 c1(C(=O)NC2C(C)CN(C(c3cnn(C4CC4(F)F)c3)=O)C2)ccc(F)c(F)c1 C1(CNC(c2oc(C3CC3)nc2C)c2n(C(CC)C)nnn2)CCS(=O)(=O)CC1 C1(NC(c2cnc(OC)nc2)=O)CC(O)CN(C(=O)CCc2nc(C)no2)C1 C(=O)(C1Cc2ccc(F)cc21)NCC1CC(NC(=O)Cc2c[nH]nc2O)C1 C1(C(=O)CN2CCC(n3cc(Cl)cn3)C2)CC2(CCC2)CO1 C1(C(N(CCCNC(C(C)SC)=O)CC2CCCC2)=O)CCN(S(C)(=O)=O)C1 c1(CCC(=O)NC2CC(C)(CNC(C(CCC)OC)=O)C2)cc(C)cc(C)c1 C(CCN=c1[nH]c(=NCCC(=O)N2CCCCC2)[nH]c2cc[nH]c12)OCC(=C)C c1(NC(C(=O)NC(N(CCS(C)(=O)=O)c2ccccc2)=O)CO)c[nH]ccc1=O Cc1ccc(C2(Cc3ccccc3OC(F)(F)F)CC2)cc1.C1(=O)CN1 CCC(C)(C)C(O)C(=O)N1CCOC(C)C1C(=O)NC1(C)CCCCCC1 C1(NC(C(C=C)(C)O)=O)CN(C(=O)COCCC2CCCC2)C2(CCC2)C1 N1(C(COCC(C)(C)C)=O)CC(NC(C2CC3(CCCO3)C2)=O)C(C)(C)C1 C(=O)(C(C)(F)c1ccccc1)NCC(C)N(C)C(C1CSCN1C)=O C#Cc1ccc(C(N2CCCC(O)(CCNC(C34CC(CO3)C4)=O)C2)=O)cc1 C(=O)(CC1=NNC(=O)C1)NCc1ccc(NC(C(C)NS(CC)(=O)=O)=O)cc1.OCC N1(C(C(C)CN2CCOCC2)=O)CCCCCC1CO N1(C(c2ccc(F)cc2)C)CCCCC(C(=O)C(N)CC#N)C1 c1(C(=O)NC2CCC(NC(=O)C(c3cccc(F)c3)O)C2)cc2ccccc2[nH]1 c1(C(N2CC3N(C(c4c(C)cccc4)=O)C3C2)=O)ccc2ncsc2c1 CC1(C)CC(CNC(c2csc(C3CC3)n2)=O)CN1C(=O)Cn1cc(CO)nn1 C1(C(N(C2CN(C(=O)C3=C(Cl)CCC3)CCC2O)C)=O)Cc2ccccc2S1 Cc1ccc(O)cc1C(N1CCC(C)C(NC(=O)CCc2ccc(C3CC3)o2)C1)=O N1(C(C(C=C)CC)=O)C2CCC1C(C(=O)N(CCCN(C)C)CC)C2 c1(C(=O)NC2C(C)(C)C(CNC(=O)Cc3cnoc3)C2)c(N)cccc1[N+](=O)[O-] c1(N2CCCC(C(=O)OC)C2)ncc(C2CCCCC2)cc1Cl N1(C(CC)=O)CCC(C)C(NC(=O)COCCc2ccc(Br)s2)C1 Cc1nn(C)c(C(=O)NC2CC(C)N(C(c3cc(Cl)ncc3N)=O)C2)c1Cl Clc1ccc(Br)c2cc(CNCCCCCOc3ccccc3)ccc12 c1(NC(C23CC(NC(c4cc(C)sc4C)=O)(C2)C3)=O)nc2ccc(Br)cn2n1 C(C(C(=O)NC1CCCC(C)C1)C(C)(C)C)NC(C1(COC)CCCC1)=O C1(C(=O)NCC2CN(C(c3c(C)noc3C(F)F)=O)CC2C)C2CC3C(C2=O)C13 C1(NC(N2CCC(CC(=O)NCC3(CCC=C)CC3)C2)=O)CC(=O)OC1(C)C N1(C(C2(CC)CC2(F)F)=O)CCC(N(C)C(c2cc(CS(C)(=O)=O)on2)=O)CC1 C1(C(C(N2CC(=CCC)C2)=O)C)CCCN(C(C2(C)CCOC2)=O)C1 C1(C(=O)Nc2c(C)cc(CC)nc2)COC2(C1)CN(C(=O)CN(C)C)C2 CCC(CC)(C(=O)N1CCC2CN(C(c3nnccc3C)=O)C2C1)C(C)C Cc1ccc(C(F)(F)F)cc1C(=O)NCC1CN(C(=O)Cc2cnsc2)CCO1 C(C)(C)(CCCN=c1nc(C2CC2)[nH]s1)NC(C(CC)NC(C)=O)=O C(=O)(C(C(C)C)NC(C1CCCOCC1)=O)N1CC(C)(CC=C)C1 c1(C(=O)NCC2(CO)CCN(C(CC3C(C)CCO3)=O)C2)nnc(O)nc1O c1(C(=O)NC(CNc2nccc(OCC)n2)(C)C)cccc2scnc12 C=CC(C)(CCOC)C(=O)N1CCN(C(c2cccc(COC)c2)=O)CC1C Cc1cc(N)c(C(=O)NC(CCNC(c2ocnc2C)=O)C(C)(C)C)nc1C C(=O)(CCC(C(C)C)NC(=O)CC1CCSC1)Nc1cncc(C#C)c1 N1(C(c2cc(Br)ccc2F)=O)CCC2C1CCCN2c1ncc2ccccc2n1 C(C(C(=O)c1ccccc1)C(C)C)NCC(C)SC C1(CC(=O)NCC(C(C)C)(C)F)N(C(C2CCCCCN2C)=O)CCC1(C)C C12(C(=O)NCCc3cn(CC)nc3)CCN(C(C3CCCCC3O)=O)CCC1C2 c1(-n2cc(C(=O)Nc3ncc(CC)s3)nn2)ccc(F)cc1F c1(OCC)ncccc1C(=O)N(CCCCCNC(c1nnn(CC)c1C)=O)C C(=O)(C(C)(C)CN1CCOCC1)N(CC(C)N(C(=O)CNC(N)=O)C)C C1(C(C)C)CN(C(c2ccc(N(C(=O)CCF)C)cc2)=O)CCCN1C(N)=O S(=O)(=O)(c1ccc(Br)cc1F)NCC1CCCN(C(C2CCC(CO)CC2)=O)C1 C1(C(=O)NC2C(CNC(CC(C)n3cccc3)=O)C2)CCCCCCC1 C1(C(=O)NCCC(=O)OCC)CC2CC2N1Cc1ccc(F)cn1.OCC C1(NC(CCSCCC)=O)CCC(C)N(C(=O)C2=COCCC2)C1 C(=O)(C1=Cc2ccccc2C1)N1C(CC(N2CCN(CC)CC2)=O)CCC1 C(=O)(C(C)CC(C)CC)NCCCN(C)Cc1c(OCC#C)nccc1 N1(C(C(COC)NC(C23CCC(CC2=O)C3)=O)=O)CCCCN(C)CC1 c1(C(N(C)CC2N(c3snc(C)n3)CCC2)=O)c(C(F)(F)F)nc2n1CCCC2 C1C(C(C)(C)C)C(=O)N1.CC1CCOCCN1Cc1ccccc1 N1(C(CCC(=O)OCC)=O)CCN(C(c2cc(F)c(CO)c(F)c2)=O)CCC1C c1(COC(C)(C)C)ccc([N+](=O)[O-])cc1F.c1(CC2C(=O)N2)ccc(O)cc1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CCC(F)(C(=O)Nc2cncc([N+](=O)[O-])c2)C1 CCCS(=O)(=O)CC(=O)NCC(C1CCOCC1)NC(=O)CCCCC=CC C(c1cccc(F)c1)=CC(=O)NCCC(C)N(C(=O)C(=Cc1cnc[nH]1)F)C c1(C(N2C(C(=O)NCCC3C(C)C3)CC(C)(C)C2)=O)ccc2c[nH]nc2c1 CC1CN(C(=O)CSc2cncc(Br)c2)CCCN1C(C1CCCO1)=O c1(C(N2CC(CNC(c3cnsn3)=O)C3C2C3)=O)n[nH]c2nccc(Cl)c12 c1(C(N2CC(N(C(CCc3cccc(OC)c3)=O)C)C2)=O)cnc2scc(C)n12 C1(C(=O)NC2CC(CCOC)C2)(NC(C23CC(F)(C2)C3)=O)CCC(C)(C)C1 C1(C)(CNC(C2(NC(C)C)CC2)=O)CCCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 c1(C(=O)NCC(=O)NCCC(C)NC(C(C)CF)=O)ccc2nn[nH]c2c1 C(N=c1[nH]c(=NCCOC2CCCCC2)[nH]c2ccsc12)C1CC2(CC=CC2)C1 C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NCCCCNC(=O)COCCCF N1(C(C(c2ccccc2)OC)=O)CCC(NC(c2ccn(C3CC3)n2)=O)C12CC2 C1(C)(C(=O)NCC(N(C(CN(S(C)(=O)=O)C)=O)C)C2CC2)CCCN1C C(C)(CCN=c1[nH]c2ccc(Br)cc2o1)NC(C1(C)C(CC)CCC1)=O Cn1[nH]c(=NC(=O)NCC(c2ccncc2)O)cc1C1CCCC1 Cc1ccc(OC(C)C(=O)NCCC2CC(NC(=O)CCOC(F)F)C2)c(C)c1 N1(CC(C)NC(=O)CNS(N)(=O)=O)CCN(C(C2CC2c2csc(=N)[nH]2)=O)CC1 S(=O)(=O)(c1ccncc1)NC1C(C)CN(C(c2cc(Br)ncc2F)=O)C1 Cc1cc(N(CCC#N)C)ncc1S(=O)(=O)CCSC(F)F C(=O)(C1CCCn2nccc21)N1CCN(C(CNC(CNS(NC)(=O)=O)=O)=O)CC1 C(=O)(CCN=c1[nH]ccs1)NCC1CN(C(C2(C)CC(F)C2)=O)CC1C(F)(F)F c1(C(=O)OCC)ccc(NC(C2(NCC3(F)CCOC3C)CCC2)=O)cn1 C=CC1(CO)CCN(C(C2C(Cc3ccccc3)CC(C)C2)=O)C1 N1(C(C2(CC=C)CCCC2)=O)CCC2CCN(C(=O)Cn3nnc(C)n3)CC2C1 c1(C(N2C3(CNC(CSCCOC)=O)CCC3CC2)=O)cnc2ccccc2n1 c1(CC)nn(C)c(CC(N2CCC(O)C(NC(=O)C=C(Cl)Cl)C2)=O)c1Cl O=C(C1=CCCSC1)NC1CCCC(NC(c2cnc(S)nc2)=O)CC1 c1(CC(N2CC(OC)C(NC(=O)COc3ccsn3)C2)=O)ccc2nn[nH]c2c1 Cn1cnnc1C(C)(C)C(=O)NCCC(O)CNC(=O)CCCNC(N)=O CCC(O)C(C)C(=O)N1CC(OCCC(=O)NCC23CC(F)(C2)C3)C1 N1(C(C2CCN(C(CCOCC#C)=O)C2)=O)CCOC(COC)C1 CC(C)C(C(=O)N1CCC=C(C(=O)NCC2C(C)(C)C2(C)C)C1)C(C)C C1(C(=O)NC(CN(C(CCOCCOC)=O)C)C)COC(C)(C)C1 c1(C(=O)NCC2(O)CCN(C(C(C)CSC(F)(F)F)=O)C2)cc2c(=O)[nH]ccn2n1 Cc1cn2c(n1)C(C)CC(C(=O)NC1CN(C(c3ccn(C(C)C)n3)=O)C1)C2 N1(C(COCCC)=O)CCC2(CN(C(=O)C3CC3)C(C)C)CCCCC12 c1(C(N2CCCC(NC(c3ccco3)=O)C2)=O)ccc(-c2ccncc2)nc1O C12(C(=O)NC3C(NC(=O)C4=NOCC4)CC3)CCCCC(=O)N1CCC2 c1(C(=O)NCC(CN(C(Cc2cc(C)no2)=O)C)O)ccc(SC(C)C)cc1 C1(CNC(Cn2c(C)nnn2)=O)CC(F)CN1C(C12COCC1C2)=O N1(C(C2(C)C(CC)CCC2)=O)CCC(C)N(C(c2ccc3occc3c2)=O)CC1 C(=O)(C1CCOc2c(F)cccc21)OCC1CC1.c1(CC(=O)N)ccccc1 C=CCC(C)(C)CC(=O)NCC(C)N(CC(F)(F)CO)C.C(C)=O CC(C)(CC(F)C(=O)NC1CC(CO)C2CC12)NC(C1C=CCCC1)=O C(=O)(C(C)(C)CC(F)(F)F)N(CC(C)NC(C1CCC(C)C1)=O)C c1(C(=O)NC2CC(NC(C(CC)CC(F)F)=O)CC2O)cnc2ccncc2c1 c1(CNC(=O)C(F)=CCN2CCCC2)cccc(NC(=O)CCc2ccoc2)c1 c1(C(N2C(C)CC(NC(C34OC(C)C(C3)C4)=O)C2)=O)ccc2nc(CO)[nH]c2c1 c1(C(=O)NC(C(C)O)CO)cc(O)nc2c1CN(C(c1ccc(=N)[nH]n1)=O)CC2 C#Cc1ccc(CNC(=O)C(C)(C)S(C)(=O)=O)cc1OC c1(C(=O)OC)ccccc1C1CCN(CC(=O)NCc2nccnc2Cl)C1 c1(OC)c(C(=O)NC2CC3C2CCN3C(c2coc(C)n2)=O)cc(Br)cc1F c1(C(N(CCNC(=O)CCN2CCCCC2)CC)=O)ccc(C#N)c(Cl)c1 N1(C(c2c(CC)cno2)=O)CCN(C(=O)CCN(C)C(C)=O)CC1CC1CC1 Cc1cc(-c2nc(-c3cc[nH]n3)nn2-c2cccc(C)c2)cc(C#N)c1 CCC(C)(O)C(=O)NCC1CCC1NC(c1ccc(CC(C)C)s1)=O Cc1ccc(C(=O)NCC2CCCCN(C(c3cnnn3C)=O)C2)cc1O C(c1c(O)ccc(Cl)c1O)=CC(=O)N(CC(C)NC(c1ccnn1C)=O)C c1(C(=O)NCC(C2CCC2)NC(Cc2c(C)ocn2)=O)nn(C)cc1Cl C(N=c1nc(NC(C)(C)CC)cc(C)[nH]1)C1CCCC(NC(CNC(C)=O)=O)C1 C1(OCCOC(C)=O)CC(=O)N(Cc2ccccc2-c2nc(C)no2)C1 O(C=CC1(O)CNC(=O)C(=O)NCC(CC(=O)N(C)C(C)C)C1=O)CC N1(C(C2N(CC)CC2)=O)CCCOC(CNC(c2[nH]c(C)c(C(=O)OC)c2C)=O)C1 O=C(C1CC=Cc2ccccc21)NC1(CO)CCN(C(=O)C(O)C2CCC2)CC1 c1(C(=O)OCC(=O)NCC(C#C)C)ccc(N2CCC(OC)C2)cc1 c1(C(N2CC(OCCNC(C(CC)C)=O)C2)=O)ccc(-c2ccncc2)cc1 c1(C(=O)NCCOCCn2cc(C(C)C)nn2)ccnc2ncccc12 C1(C)(C(=O)NCc2c(C(=O)NC(c3ncccn3)C)c[nH]n2)CC(F)(F)C1 CC1CC(C(c2nnnn2CCCF)NCC2(CO)CCCCC2)CCO1 C12(C(=O)NCCCNC(C)=O)CC1CN(C(C1CCC(CO)CC1)=O)C2 Cc1cc(C(=O)N(C)C)sc1-c1ccc(N(C)CCC2CC2)cc1 C(C1CCN(C(c2cnc3n2CCC3)=O)CC1)=CC(=O)NC1CC2OC1C1CC21 c1(C(=O)NC2CCN(C(c3ccc(OC(C)=O)cc3)=O)C2)cccc2ccnn12 C(=O)(CCS(=O)(=O)CCC(F)(F)F)NC1CCN(C(C(C(C)C)O)=O)C1 c1(OC)cccc(-n2cc(CCNC(=O)OCC(C)(C)C)nn2)c1 C1(CC(=O)NCCCC(C)NC(C2(C(N)=O)CCC2)=O)CCC12CCC2 N1(C(c2cnn(C3CCC3)c2)=O)CC2(C1)CN(C(c1cc(Cl)nc(Cl)c1)=O)C2 c1(C(=O)NCCc2nnco2)ncncc1Cl Cc1c(O)c(=O)ccn1CC(=O)NC(C)CN(C)C(c1ccccc1CC#N)=O N1(C(C(n2cc(C3(SC)CCC3)nn2)C)=O)CCN(C)CC1C(C)OC C1(C(N2CC(C)(NC(=O)CN3CCCC3CO)C2)=O)CC2C=CCC(C1)C2 N1(C(Cc2cnc(C)[nH]2)=O)CC2(C1)CN(C(c1coc(C(F)(F)F)n1)=O)CCO2 c1(CC(N2CC(CC(C)NC(=O)COCCN(C)C)C2)=O)ccn(C)n1 CC1(C)CN(C(c2ncnc(O)c2Cl)=O)CCC1NC(C1CC(C2CC2)=NO1)=O C1(C(=O)NCc2nn(Cc3ccccc3)cc2Br)CCN2CCOSCC12 c1(C(=O)NCC2(C(=O)NCC3N(C(C)C)CCC3)CCCC2)occ2c1CCC2 CC(CCCC(=O)Nc1ccccc1OC(F)(F)F)NCC1CCCS(=O)(=O)C1 c1(C(N2CC(O)CC(NC(c3c(CC)scc3)=O)C2)=O)nc(C)c(C)nc1O C(=O)(C1CCCc2ccnn21)N1CCN(C(C=Cc2c(C)nccc2)=O)C(C)C1 c1(C(=O)NCCN(C)C(c2cnnc(O)c2)=O)ccc(OCC(F)F)cc1 C1(CNC(c2c(C)cco2)=O)CN(C(c2sccc2-n2ccnn2)=O)CCC1C c1(C(C)C(=O)NC2CCN(C(=O)CCc3ccncn3)C2C)nc(Cl)ccc1Cl Cc1c(F)ccc(C(N2CCC(C)C2CNC(c2cnccn2)=O)=O)c1O C(CC(C(C)C)NC(c1cncn1C(C)C)=O)N(C(c1n(CC)ccn1)=O)C C1(NC(c2cnc(C)s2)=O)CN(C(=O)Cc2ccn(CC(C)C)n2)CC(C)(C)C1 C12(OC)CCN(CC1)C2.c1(NC(c2cncc(C)n2)=O)nccc(C#N)n1 C=CC1(C(=O)N(C)CCOCCNC(C2(c3n[nH]cc3C)CC2)=O)CCC1 C(=O)(CCCCCS(N)(=O)=O)NC1C(CN(C)C)CCCC1 c1(CC(=O)NC2C(C)CN(C(=O)C(C)(C)F)C2)ccc2c(c1)CCO2 c1(OCC)ncc(C(=O)NCC(C)(O)CNC(=O)Cn2nnc(=O)[nH]2)s1 N1(C(c2nc(C(=O)OC)sc2)=O)CCC2CC1CN2C(=O)C(C)c1cccs1 C(CCCCC(=O)NCC1COC(=O)C1)n1cc(CNC(C)=O)nn1 c1(C(=O)NCCC2(C)CCN(C(C(C)CO)=O)C2)ccc(Cl)c(F)c1F N1(C(C(c2cccc(F)c2)C)=O)CCOC(CNC(C2CC2(F)F)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CCCC(CNC(c2c(C(=O)OC)scn2)=O)C1 C(=O)(CCC(C)(C)C#N)NC(CNC(c1n(C(C)C)ccc1)=O)(C)CO CN1CCN(C(=O)CCNC(c2cnc(Cl)n2C)=O)C(CO)C1 c1(CC)nc(C(=O)NC2(CNC(C3CC(C)(C)C3)=O)CCC2)co1 C12(NC(C(CO)N(C)C)=O)CCCC1N(C(c1ccc3c(c1)OCO3)=O)CC2 C(CCCCC(=O)N1CCCC(CO)(NC(=O)C=CC2CCCO2)C1)SC c1(C(=O)Nc2ccc(NS(N)(=O)=O)cc2)cc2c(cc1F)NCCC2 C(C(CC(C)C)NC(C1CCC(=O)N1)=O)NC(CC(C)OC)=O N1(C(C(CCC(C)C)NC(C2CC3(CC3)CO2)=O)=O)CCC2(CCCCO2)C1 C(C1CN(C(C2(CCOC)CCC2)=O)CC1C(=O)NCCCc1cn[nH]c1)=CC C1(NC(c2nccc(OC)c2)=O)CCN(C(c2ccc(Cl)cc2C)=O)CC1CO CCCC(CNC(C1(C)CC(F)(F)C1)=O)C(=O)N1CC(N=[N+]=[N-])C1 C(c1cccc(F)c1Cl)=CC(=O)NCC(n1cc(-c2nccc(C)n2)nn1)C C1(NC(c2nncc(OC)c2)=O)CCN(C(c2snc(C)c2N)=O)CC1CO c1(CC(=O)N(C2CCC(NC(c3cnn(C(C)C)n3)=O)C2)C)cccc(F)c1F C1(CN(C(=O)Cc2ccc(C)s2)C)CCCCN1C(c1[nH]ccc1C)=O.CCOC C1(CC)CC(O)CN1C(=O)C(CNC(C1(OC)CCCOC1)=O)CC1CCCC1 C1(COC(CC2(C)CC2(Cl)Cl)=O)CN(Cc2ccccc2)CC1C#N C1(NC(c2c(C)cn(C)c2)=O)CC2CCC1CC2NC(c1cnoc1C(C)C)=O C1(CC)CC(CC(N2CC(CC(C)(C)CNC(=O)C(O)C3CCC3)C2)=O)CCO1 N1(C(C(c2cn(CC)nc2)=O)=O)CC(CNC(=O)C2CC2)N2CCC1C2 N1(C(C2=CCN(C(C(c3ccc(C)o3)C)=O)C2)=O)CCN(C)C2(CCC2)C1 C1(NC(c2ccc(OC)c(Cl)n2)=O)CN(C(=O)C(C)(C)N(C)C)CC2CCCC12 C1(NC(C2CCOCC2)C)CCCN(C(c2cccc(-c3nnc(C)o3)c2)C)C1 c1(C(C(=O)NC2CC2)N(C)CC2C=CCC2)ccnn1C CC1(NC(=O)C2=CS(=O)CC2)CCCN(C(c2cc[nH]n2)=O)C1 Cc1ncn2ccc(C(=O)Nc3ccc(Cl)cc3C(C)(C)C)cc12 N1(C(=O)C2CC2)CCCC(C(N2CCC(n3cncn3)C2)=O)C1 N1(C(C2(C)CCNC2=O)=O)CCCc2c(F)cc(Br)cc21 c1(NCCCC(CC)O)cc(Br)ccc1S(=O)(=O)NCC1CCSC1 C12C(C)CCCN1C2.C=CC(C(=O)OC)CC C1(N(C(=O)CNC=O)C)CCCCN(C(C2(O)CC2(C)C)=O)C1 C1(CNC(c2cnc(C(F)(F)F)s2)=O)CN(Cc2ccccc2F)CCC1(F)F C1(C(N(C(C)CC(F)(F)F)C)=O)CN(C(=O)CN(C)C)CCC1(C)C C1(CNC(C2N(C(CNC(C(CC)CC)=O)=O)CC(F)C2)=O)CC2(CCC2)CO1 c1(NC(c2ccc(OC)cc2F)c2nnnn2C)cc(O)c(F)cc1F c1(C(=O)NCC2CC(NC(CC(=O)N(C)C)=O)C2(C)C)nnn2c1COCC2 C(=O)(CC(C(F)F)NC(=O)CCC(C)C)N1CCC(CC(C)C)(CO)C1 C1(C(=O)NC(CC)CO)(CO)CCN(C(=O)C(=O)N(C)C)C1 N1(C(=O)Cc2cnc(O)nc2O)CCC2(C1)CN(C(C1COC1)=O)CCO2 N1(C(CN2CCC(OC)C2)=O)CC(C)(C)C1C(C)C.C1(CN(C)C)C(=O)N1 C1(O)(CNC(c2c(C)nc[nH]2)=O)CCN(C(=O)CCc2cnccn2)C1 C(c1ccc(C)nc1)=CC(=O)N(C)CC1CCN(C(C(CC2CCC2)OC)=O)C1 CCC(CC(=O)N1CC2CCCC2C1C(N1CC(C)(C)OCC1CC)=O)C(C)(C)C c1(C(=O)NC2CCCC2CNC(c2cc(CF)on2)=O)cnc(O)c([N+](=O)[O-])c1 c1(CCC(=O)NC(C)CCCNC(=O)CN2CCOCC2)cc2ccccc2[nH]1 c1(CCCC)cccc(C(=O)NCC(C)CNC(=O)C(O)C2CC2)c1 C1(C(N2CC(N(CC=C)C)C2)=O)CCCC(NC(C2OCCC2(C)C)=O)CC1 c1(C(=O)NC(C(=O)OC)CCF)ccc(CNC(=O)CCOCC(C)C)cc1 Cn1ccc(=O)c2cc(NC(=O)Nc3ccc(CC#N)cc3F)ccc12 C(=O)(C(C)(C)CCC(=O)OC)NC(C1OCCN(C(C(CC=C)(C)C)=O)C1)C Cc1nccn1CCC(=O)NCC1(C(=O)NCCCO)CCC1 C1(CNC(C2CCC(C)(C)CC2)=O)CC(C)(C)CCC1NC(=O)CC(F)F N1(C(=O)OC(C)(C)C)CC2CC(NCCc3cc(OC(F)F)ccc3F)CC1C2 c1(CC)nocc1C(=O)NCC1CCN(C(=O)C(C)(C2CC2)NC(C)=O)C1 c1(C(C)(C)C)ccc(C(=O)NC(c2ccc(Cl)cc2)C(F)(F)F)c(F)c1 CCN=c1ccc(C(=O)N(C2CCCN(C(c3cnco3)=O)C2)C)c[nH]1 C1(C(N2CCC3C(NC(c4cnc(SC)n4C)=O)C32)=O)CCC(=O)N(C)C1 N1(C(c2ccc(C)nc2)=O)CC2CCC1CC2NC(=O)CC1=CCOCC1 CCCC(CC1CCCC1)C(=O)NC1CC(CNC(C2CC3(C2)CC3(F)F)=O)C1 N1(C(C2(OC(C)C)CCC2)=O)CC(CNC(=O)C(C#N)C(C)C)C2(CC2)C1 CC1CCC(C(N2CC(C)C(F)(F)C2)=O)CN1C(=O)CSCC(F)F O=C(CC1C(=O)Nc2ccccc21)NCCC1(O)CN(C(C2(O)CCC2)=O)C1 C(=O)(CCCCCC#N)N(C1CCCCN(C(c2ccccc2C(F)F)=O)C1)C O=C1CCCC(C(N2CCCCC2C(=O)NCC2CCNC(=O)C2)=O)CC1 c1(C(c2n(CCC)nnn2)NC(C)C(=O)NCCOC)cc(Cl)sc1C C(=O)(C(C#N)C(C)(C)C)NC1(C)CCCN(C(c2cc(OC)c(O)nc2)=O)C1 c1(C(N2CCC(CNC(CCc3scc(C)n3)=O)CC2)=O)sc(C)c(C)c1C N1(C(CSCc2nc(C)[nH]n2)=O)CC(NC(c2cc(C(N)=O)n(C)c2)=O)CC(O)C1 N1(C(C(CCC)OC)=O)CCN(C(c2cc(=O)c(OC)co2)=O)C(COC)C1 c1(C(=O)NC2(C)CC(NC(=O)C(N)=O)C2)ccn2c(Br)cnc2c1 n1(CCC(=O)NCC(CNC(C(C)OCC=C)=O)(C)C)nc(C)c([N+](=O)[O-])c1C N1(C(c2nc(C(C)(F)F)sc2)=O)CC2CCN(C(C3CCCCCC3)=O)CC2C1 C1(OCC(N2C(CNC(c3cc(C(CC)CC)no3)=O)CC2)=O)CCC(C)CC1 C=C1CCCN(C(C2(C(C)NC(=O)C(C3CCCCC3)F)CC2)=O)C1 c1(C(N2CCN(C(C3CC(C)OC3=O)=O)CC2)=O)cncc2c1CCC2 N1(c2cc(C)nc(Cl)n2)CCC(NC(=O)Cc2nocc2C)C(C)(C)C1 c1(C(=O)NCC(CO)NC(=O)Cc2cncs2)cccc2c1COCCN2 c1(CNC(c2n(C(C)C)nc(C(C)C)c2)=O)cc(Br)cc(F)c1O.N12CC(C1)C2 CCC(C)CCCC(=O)NCC(C)(C1CC1)NC(CC=CC)=O N1(CCc2cccc(C)n2)CCC2(CC1)CC2NC(=O)Cc1cccc(F)c1O CCCC(C(=O)NCCCOCCCO)NC(=O)C(C)n1ccnn1 C1(C(C)C)C(NC(c2coc(O)n2)=O)CCN1C(=O)COc1ccc(O)cc1 CC(C)CCC(O)C(=O)NCC1CN(C(c2ocnc2C2CC2)=O)CCC1(C)C N1(C(C2(C(C)NC(c3cc(C#N)c[nH]3)=O)CC2)=O)CCOC(C)(C)C1 C12(NC(c3c(C)cccc3C)=O)CCC(NC(C3CCOCC3)=O)(CC1)CC2 c1(NC(=O)C(=O)NC2CCN(C(=O)CNS(=O)(=O)C(F)F)C2)ccc(Cl)cn1 n1(C(C)C)nc(C(F)(F)F)cc1C(=O)NCC1CCN1C(C1CCCCO1)=O C(CS(=O)(=O)CC(=O)NC1CC(CNC(=O)C(C)C(C)C)C1)OC C(=O)(CCCCc1cnn[nH]1)NCC1CC(NC(C2C(F)(C(=O)OC)C2)=O)C1 c1(CC(=O)NC2(C)CCN(C(C3CCN(C(C)=O)C3)=O)C2)ccc2ocnc2c1 CC(C)CCC(O)C(=O)N1C(C)CC2CNCC12 Cc1csc(=NCC(=O)NC(CNC(=O)C(O)C2CCC2)C(C)C)[nH]1 n1(CC)c(C)nn(CC(=O)OCCCNC(=O)C(C(=O)OC)N(C)C)c1=O C1(NC(C(CC)C)=O)CC2CC1N(C(=O)CCCCOC)C2 n1(CC(=O)NCCN(C(C(C)n2ccnc2)=O)C)cccc1CC(=O)N(C)C c1(NC)scnc1C(=O)NCC(C)(O)CNC(=O)CNS(N)(=O)=O C#CC1(O)CC(C(=O)N(CCCCN(C)C(C2(C(C)(C)C)CCCCC2)=O)C)C1 C1(N(CC(C)C)C(=O)CN2CC(=O)NC2=O)CCCN(C(=O)CCCCN(C)C)C1 CC1(NC(C2C3CN(C(C45CCC(C4)C5(C)C)=O)CC32)=O)CC2CCC(C1)S2 c1(CC(=O)NC2(CCCNC(c3c(CCC)n[nH]c3)=O)CC2)ccc(F)cc1 C(N=c1[nH]c(=NCCS(=O)(=O)CCOC)c2cccc(F)c2[nH]1)C1(CO)C(C=C)C1 O=C(C#CC1CC1)NC1CC(CC(=O)NCCc2ccccc2Br)C1 C1(CC)CCCN(C(=O)CC(C)CN(C)C)C1C(=O)NC(c1cccnc1)CC CC12CCC(CC1)NC(=O)C1(CC1)CNC2.c1(CCNC(=O)CO)cccs1.CO Cn1ccc2sc(C(N3CCC(F)C(NC(=O)C=CC(C)(C)C)C3)=O)cc12 S(=O)(=O)(CCC=O)NC.C(CC(=O)NCCCNC(=O)C(C)C)SCC C(=O)(CC(CNC(c1nc(NC(=O)OC(C)(C)C)sc1C)=O)C(F)F)OCC C(C(C)CN=c1cc(-c2cc(C)ccc2F)nc[nH]1)NC(CSC)=O c1(N(C)C)ccc(CNC2CCN(C(=O)NC(=O)C(Cl)(Cl)Cl)C2)c(Cl)c1 C(CC(F)F)(C(=O)NCc1ccc(O)nn1)NC(=O)CC1(O)CCCOC1 C12(CNC(C(CNC(c3c(CC)con3)=O)N(C)C)=O)CCC(CC1O)C2 N(C(=NCC1CCCOC1)N1CCC=C(c2ccco2)C1)C1CCS(=O)(=O)C1 C1(NC(c2ccc(C(F)F)cc2)=O)CCN(C(=O)Cn2cccc2)C12CC2 C1(C(=O)NC2(C3CCCN3C(=O)C(=Cc3c[nH]cn3)F)CC2)CC2(C1)CC2F c1(C(N(CCCN(C(=O)CCOc2ccc(F)nc2)C)C)=O)[nH]cc2c1CCC2 c1(C(C(=O)N(CC(n2cc(C(CSCC)C)nn2)C)CC)F)cccc(C)c1 Cc1ccc(C)c(N(CCCNC(=O)C(Cc2cnn(C)c2)CN)C)c1 C1(N(C(C2(OC)CC2)=O)C)CCN(C(=O)C(C)(C)N2CCCCC2)C1 c1(NCC(CNS(CC)(=O)=O)O)ccc(S(=O)(=O)NS(=O)(=O)CC2CC2)cc1F Cc1cccc(CCNC(C2CC(C)N2C(=O)CC2CCCC2O)=O)c1 N1(C(=O)CCc2cccc(Cl)c2)CCN(C(c2cc(O)ncn2)=O)C2CCC12 N1(C(C2CCN(C)S2(=O)=O)=O)CCCN(c2ccccc2)CC1(C)C CC1=CCN(C(=O)C(C)(C2CCC2)NC(c2c[nH]c(=N)o2)=O)C1 C=CCC(C(=O)NC(CNC(=O)CN(C)C(=O)OC(C)(C)C)C1CC1)C(C)(C)C c1(OC)ccc(O)cc1NC(=O)CN(C(c1cncc(C)n1)=O)C(C)C c1(C(=O)NC2(C(=O)NCC(F)C3CCC3)CCN(C)C2)ncc2ccccn12 c1(C(N2C(CCN(C(CCCCC)=O)C)CCCC2)=O)c[nH]c2cccnc12 c1(C(C(=O)NCCOCC)N2CCC2CC)ccc(OC(F)F)cc1 C1(C(=O)OC2C(NCC=C)CCC2)(CC)CCCCCC1 C1(NC(=O)Cn2cnnn2)CCC(NC(c2cnc(C3CCC3)o2)=O)CC1 N1(C(C2(C3CCCO3)CCCC2)=O)CCCCC1Cc1ccccc1Br C12(C(N(C3CCCCC3)CC#C)=O)CCCC1CN(C(=O)CCS(N)(=O)=O)C2 c1(C(N(CC(CC)NC(=O)C(C)SC)C)=O)ccc(F)cc1-c1cccs1 C(=O)(C1CCCc2ccnn21)NCC(C1CCCCC1)NC(C1OCCN(C)C1)=O N(C(=NCCc1ccco1)NCC(c1ccccc1)F)Cc1n(C)ncc1 N1(C(C=CC(CC)C)=O)C2CCC1CC(NC(c1cccc(Cl)c1C)=O)C2 C(C)(C)(C(=O)NCc1ccc(C(=O)NC(c2ncc(C)s2)C)s1)OC(C)=O C(C)(CCCC(=O)N1CC(N2CC(O)C2)C1)NC(C(C)N(C(C)=O)C)=O c1(C(=O)NCCN(C(=O)CC2C=CS(=O)(=O)C2)CC)cccnc1-n1ccnc1 Cc1cc(C(=O)NC2(C)CC(NC(=O)C(C)C(O)C(C)C)C2)c(O)cc1F c1(CNC(C2C(NC(=O)OC(C)(C)C)C3CCC2C3)=O)ccc2[nH]ccc2c1 N1(C(C(C=C)(F)F)=O)CCC(C)(C)C(C(=O)NCCN2CCOCC2C)C1 c1(OC)ccc(F)c(C(F)(F)F)c1Cl.N12C(=O)CCC(C1=O)C(=O)C2 C1(NC(C(C)NC=O)=O)CC2CCC1N(C(c1ccn(C)n1)=O)C2 n1(CC(=O)NC(CCNC(C2C(C)C2)=O)(C)C)ncc2ccccc12 N1(C(C(C)OCCC#C)=O)CCCCC2(C1)CN(C(=O)C=C(Cl)Cl)C2 c1(C(=O)NCC(C(C)C)NC(c2cccc(CC)n2)=O)cnc(OC)c(Cl)c1 c1(OC)cnc(C(N2CCOC(C(C)NC(=O)CC(C)O)C2)=O)c(F)c1 CCCCC(CN=c1nc(SC)[nH]cc1C)NC(=O)COc1cccc(CC)c1 N1(CCCNC(c2ncc(-c3c(C)cccc3)o2)=O)C(=O)c2ccccc2C1=O C1(CCNC(c2c(C)nc(C3CC3)s2)=O)CC(F)(F)CN1C(=O)C1=CCCC1C N1(C(C)C)N=C(C(=O)NC2C=CCN(C(c3cc(O)n(C)n3)=O)C2)CCC1=O C(=O)(CCCCC(C)(C)OC)NC(c1c(OC)cccc1)C(C)SC C1(C(=O)NCCC(C)NC(c2cc[nH]n2)=O)CC(=O)N(C2CCCCC2)C1 N1(Cc2c(Br)ccc(OC)c2)CC2CCN(C(c3cccn4cncc34)=O)C2C1 C12(C(=O)NCC3(O)CC(NC(c4ccccc4)=O)C3)CC3CC(CC1C3)C2 CCC(C)C(O)C(=O)N(C)CCOCCN(C(=O)CN1CCCC(C(N)=O)C1)C N1(CC)CCOC(CNC(=O)CC2(N(C(=O)Cc3coc(C4CC4)n3)C)CC2)C1 c1(C(=O)NC2(CNC(C(C)OC)=O)CCOC2)ccc(C(C)CC)nc1O CC1(C(=O)NCc2ccnc(F)c2)CC12CCN(C(CCC(=O)O)C(=O)O)CC2 C1(C(=O)NC2CCN(C(=O)CCOC3CCC3)CC2O)CCn2c(O)nnc2C1 N1(C(c2c(C)ncn2O)=O)CC2CCC2(CNC(c2c(F)cncc2Br)=O)C1 CCCCCCCC(=O)NCC1(NC(c2ccn(C)c(=O)c2)=O)CCCCC1 CC(CC(=O)N1CCC(CNC(=O)C(C)(C)n2cncn2)C1)n1ccnc1 c1(OC)ccccc1C(C)C(=O)NC1CC(CO)N(C(C2CC(=C3CC3)C2)=O)C1 CC1(C(=O)NCC2CC3CN(C(=O)C=C4CCC4)CC23)C2Cc3ccccc3C12 c1(C(C(=O)NCC(=C)CCNC(=O)C=CC(=O)N(C)C)C)c(Cl)cccc1Cl Cc1[nH]c(C)c(C(=O)NCCC(C)(C)C(=O)NC2(C)CCCC2(F)F)c1C c1(C(C)=O)cc(C(=O)NCC2(F)CC(NC(=O)COc3ccccc3)C2)oc1C c1(NC(C(C2N(C(C(CC)OCC)=O)CCC2)(C)C)=O)ccc(F)c(CO)c1 c1(NCC2C(C)CN(C(=O)Cc3c(Cl)cccc3Cl)CC2)ccnc2ncnn12 c1(N(C)CC2C(C)C2)nc(NCCc2nc(=N)[nH][nH]2)c2ncn(C)c2n1 CC1CN(C(=O)C2CC2)CC1NC(=O)N(c1ccccc1Cl)C1CC(=O)N1 C(=O)(C(C#N)C(C)C)N(C)CC1N(C(c2cc(C)nn2C(F)F)=O)CCC1 C(=O)(C(CCCC#N)N1CCN(C)C2CC12)Nc1c(C)cccc1 C1(CNC(CCOC)=O)CC(OC)CN1C(c1ccc(C2CCC2)nc1)=O N1(C(c2cc(COC)[nH]n2)=O)CCC(NC(=O)CCF)C1(C)C N1(C(c2cc(C)n(C(C)C)n2)=O)CCCC2(C1)CN(C(=O)CCC1CCOC1)C2 C1(NC(CC2(CC)CC2)=O)CN(C(c2cc(C3CC3)ncn2)=O)CCC12CCC2 c1(CC(N2C(C(=O)Nc3c(C(N)=O)nccc3)CC2)=O)cccc([N+](=O)[O-])c1 S(=O)(=O)(c1ccc(F)c(C)c1)N1C(C(=O)Nc2cnc(OC)nc2C)CC(F)C1 c1(C(N2C(C(=O)NCCCOCC)CC2C)=O)cc(C)ncn1.NCC CC(O)CCCCCC(=O)N1CCN(C(C2(C)CCCO2)=O)C2(CC2)C1 c1(N2C(CCNC(CS(CC)=O)=O)CCCC2)cccc(F)c1[N+](=O)[O-] c1(NC(=O)NCCn2nccc2Br)cnc(N2CCCCC2)nc1 N1(C(c2n(CC#C)cnn2)=O)CCN(C(=O)Cn2nccc2C)C(CCO)C1 C1(C)(C(N(C2CC(C(N)=O)C2)C)=O)CN(C(=O)CCC(CF)CF)C(C)(C)C1 c1(C(=O)NCC=CCNC(C2C(C#C)C2)=O)cccc2ncsc12 c1(OC)c(N2CCC(C)C(NC(C3CCC4CC4C3)=O)C2)ncnc1C C12(CNC(CNC(N)=O)=O)COC(CNC(=O)CCc3nccs3)(C1)C2 Cc1nn(CCO)c(C)c1C(=O)NCC1CCCC1NC(C1(C)CC=CCC1)=O N1(C(C2(OC)CCCC2)=O)CC2C(CNC(C3CCCN3C=O)=O)C2C1 Cc1nncc(CNC(=O)N(C)CC2CNC(=O)N2)c1C c1(OC)ccc(Cl)c(C(=O)NC2CC(N(C)C(c3cc(Cl)n(C)n3)=O)C2)c1F N1(C(C=C(C)C(N2CCCC2C=CC2CC2)=O)=O)CCCC(C)(C#N)C1 c1(OC)ccc(F)c(C(N2CC3CC2C3CNC(C2CCCSC2)=O)=O)c1N c1(C(=O)NCCC2N(C(CCCC)=O)CCCC2)cc([N+](=O)[O-])ccc1SC C(=O)(CCCCCF)N1C(C)CC(NC(C(C)Cc2ccccc2F)=O)C1 C1(O)(C(N2CCC(C(=O)OCC)C2)=O)CCN(Cc2cc(OC)ccc2Cl)CC1 CCCCCCC(CC)C(=O)NCCCC1CCCN1C(C1CC2(CSC2)C1)=O C(C(CC)(CC)C(=O)NCc1cccnc1)NC(C1N(CC)CCC1)=O C12(CNC(C(C)C3CCCO3)=O)CN(C(=O)CCc3ccc(N)cn3)CC1CCO2 c1(C(N(C(C)C)C2CC2)=O)cc(CNC(C2CCCC2F)=O)nn1C CC1(C)CC(C(=O)NC2CC2CNC(c2cc(N)c(F)cc2F)=O)CC1(C)C c1(OC)cccc(F)c1CN1CCSCC1C(=O)N(CCC(C)CO)C1CC1 c1(CC(=O)NC(C2CN(C(C3CCCS(=O)(=O)N3)=O)C2)C)cn2ccccc2n1 c1(CN(C(c2coc(CSCc3ccccc3)c2)=O)CC)ccc(C)c(C#N)c1 C(=O)(CN=c1[nH]c(=NCCCSC)c2ccccc2[nH]1)N(CC)CC C1(c2nnc(C(N(CCN(C)C)C)=O)o2)Cc2ccccc2C1 C(=O)(C1CCOc2ccccc21)N1CC(NC(c2c(C(C)C)occ2)=O)C(C)C1 c1(OCC(=O)NC2CCC(NC(c3c(CC)oc(C)c3)=O)C2)ccc(C)cc1C c1(C(N2CC(CC(=O)NCC3CC(O)C(O)C3)(OC)C2)=O)ccc(O)nn1 C(=O)(CCS(=O)(=O)N1CCCCC1)NC1C(NC(CSC)=O)CCCC1 CON1CCC(C(N2CC(OCC(=O)NCCN=S(C)(C)=O)C2)=O)CC1 c1(C(=O)NC2C(CNC(C3CC(OC)C3)=O)CC2)ccc(-n2ccnn2)cc1 Cc1nc(NC(C2CC2C(=O)Nc2nccc(Br)c2Cl)=O)c(C#N)n1C C1(C2CCC2)(C(N2CCC(CN(C(C3C(CC)OCC3)=O)C)CC2)=O)CCC1 CC1CN(C(C2(CO)CCN(C(=O)Cn3ncn(C)c3=O)C2)=O)CCCO1 C(=O)(CCCn1cccc1)N(CC(c1ccccc1)c1ccccc1)C(C)C CC(C)C1=NOC(C(=O)NCCC(C)N(C)C(c2cc(O)cc(=O)o2)=O)C1 CC1CCCC(CCNC(=O)CC2CCCC2NC(C2(C(F)F)CC2)=O)C1 Cc1cc(C(=O)N(CC(C)CNC(C2(SC)CC(O)C2)=O)C)cc(O)n1 c1(NC(=O)Cc2ccc(OCF)cc2)cn2ccc(-c3ccc(F)cn3)cc2n1 C(=O)(CN=S(C)(C)=O)NCCCN(C(c1ccc(C(=O)NC)nc1)=O)C1CC1 N1(C(c2cc(C)c(C)s2)=O)CC2(CC(C(=O)NCCOC3CCC3)CO2)C1 N1(C(=O)NCC(c2ccc(C)c(C)c2)O)CCCCC12CCOC2 C1(NC(C(c2ccccn2)C)=O)CC(C)N(C(=O)C=CC2CCOCC2)C1 c1(OCCC(=O)NC2CN(C(=O)COCC(=O)NC3CC3)C2)ccccc1F c1(C(=O)OC)sc(NC2CCC(NC(C3CCC(C)CC3)=O)CC2)nc1Cl C1(C(=O)NCCC2(OCC)CCC2)CC2(C1)CC(C#N)C2.C1(=O)CCN1 N1(C(C2CCC(C(N(C)Cc3ccc(C)[nH]3)=O)CC2)=O)CC2CCC(C1)N2C C(CCCCCCO)NC(=O)NCC1CC12CCCCC2 c1(C(=O)OC)nccnc1NCC(C1CCOC1)NC(=O)CC1CCCCC1 C(C(CC(F)(F)F)NC(=O)Cn1nccn1)NC(C1N(C)CC1)=O c1(C(=O)NCCCN(C)C(C2CN(C)CCN2C)=O)cccc(O)c1F Cc1cccc(Cl)c1C(=O)NC1CCN(Cc2cccc(C)c2Cl)CC1F N1(C(=O)OCC)CCN2CC3(CC3)CC2C1.c1(CC)cnc(CNC(=O)COCC)s1.C1CO1 CCC(CC(=O)N1CC(C(C)NC(C2CC(O)CN2C(C)=O)=O)C1)OC Cc1cc(=O)oc(C)c1C(N1CC2CC2(NC(C2CCCN2S(C)(=O)=O)=O)C1)=O c1(CC(=O)NC2C(CNC(C(F)=CCC)=O)CCCC2)c(C)nc(CC)nc1C c1(C(=O)NCCC2CCCN(C(c3cn(C)nc3)=O)C2)cc(N)c(Cl)c(O)c1 C(N=c1nc2c(c[nH]1)COC2)C1(CNC(C2CCCC(C)C2)=O)CC1 c1(CCC(=O)NCC(CC=C)NC(=O)C(N)=O)cc(Br)ccc1C N#CC1(C(N2C3CCC(C3)C2C(=O)NC2COC3(CCCC3)C2)=O)CCOCC1 c1(C(=O)NCC(CNC(C(C=C)O)=O)C)c(F)c(C)cc(N)c1F c1(N(CC(=O)N(c2c(CN3CCSC3)cccc2Br)C)C)c(O)cccc1C#N.CO c1(OC)ccc(C(=O)NCC23CC2CN(C(=O)CN2CCC(C)C2)C3)cn1 C1(C(N(C)CC2OCCN(C)C2)=O)CN(C(c2ncc(F)cn2)=O)CC1(C)C c1(C(=O)NC2(C)CN(C(=O)Cc3c[nH]c(=N)nc3O)C2)ccc2nccn2c1 C12(C(=O)NCCC3N(C(CCC=CC)=O)CCC3)CCC(N=[N+]=[N-])C1C2 N1(C(CSc2nc(C)[nH]n2)=O)C2CCC1CC(CNC(C1COCCO1)=O)C2 C(=O)(C#CC1(C(F)(F)F)CC1)NC1CCCN(C(c2cc(C)sc2C)=O)C1 C1(CNC(CC(=O)NCC)=O)CCC12CN(C(=O)CC(c1c(C)noc1C)C)C2 C1(CC(=O)NC(C2CN(C(C(C)Cc3ccco3)=O)C2)C)CC=CCN1C c1(C(=O)NC2(CNC(c3c[nH]c(=NC)o3)=O)CCCCC2)[nH]cc2c1CCCC2 Nc1ccc(C(N2CC3CCN(C(=O)CCSC(F)(F)F)C3C2)=O)c2c1CCCC2 CCC(F)(F)C(=O)NCC(C1CCC1)NC(C1(C)CCCO1)=O N1(C(c2c(OC)cc(O)cc2)=O)CC(NC(=O)CC(C)O)C2(CCC2)C1 N1(C(C(=O)NC(c2cc(C)ccc2C)CC)=O)CCC2CC(C(=O)OCC)C2C1 c1(C(N(C2CCN(C(=O)C(C)c3ccon3)C2)CCC)=O)ccnn(C)c1=O c1(C(c2nnnn2CCCOCC2CC2)NS(C)(=O)=O)cc(Br)ccc1F c1(C(N2CCCC(F)C2)=O)cc2c(C(F)(F)F)cccc2s1 N1(S(c2cccc(C(=O)OC)n2)(=O)=O)CC(C)Oc2cc(F)ccc21 C(=O)(C1Cc2c(Cl)cccc21)N1CCCC(CN(C(C2CCC(CC)O2)=O)C)C1 Cc1nc(Cl)cc(Cl)c1C(N1CCCC1(C)C(=O)Nc1c(Br)ccc(F)c1F)=O N1(C(C2CC(=C)CN2C(C2CC2C(=O)OC)=O)=O)CCc2cc(F)ccc2C1 Cc1cc(O)cc(=O)n1CC(=O)NC1CN(C(C2CC2C#N)=O)CC1C1CC1 N1(CCOCCC(=O)NC(N)=O)CCCN(C(=O)CSCC(=O)OC)CC1.CO c1(C(N2CCC(CN(C(=O)C3=CCS(=O)(=O)C3)C)CC2)=O)ccc(S(N)(=O)=O)o1 C(C(=O)NC(C)C)(C1=CCSC1(C)C)N(C)Cc1cnc(CC)s1 c1(NC(COC)CC)ncnc(NCC(c2ccccc2)C)c1C c1(C(N2C(CCC(N3CC(C)C(=O)CC3)=O)CCC2)=O)ccc2c(c1)nnn2C CC(O)C(C)(C)CNC(=O)C(C1CCCN(C(C2CCC(C)(C)C2)=O)C1)(C)C Cc1csc(C(N2CCCCC2c2ccco2)C(=O)NCC2COC2)c1C N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CC(NC(=O)C=CC3CC3)CC2C1 C12(NC(CCCn3ncn(C)c3=O)=O)CC3CCC(C1C2)N3C(=O)CO CC(C)CC(C(=O)NC1CC2(CC2)CO1)ONC(=O)CNC1CC(C)C1 N1(C(=O)OC)CCC2(CC1)CC2NC(=O)C(F)C1CC(CNc2ocnc2C)C1 c1(C(=O)NCCn2cc(-c3cc(OCC)cc(F)c3)nn2)cc2nc[nH]c2cn1 Cc1nc(C)c(C(=O)NC2CCCC(C(=O)NC3(c4cccc(F)c4)CC3)C2)[nH]1 C1(C(N2C(C3(C(=O)NC(C=C)C4CC4)CC3)CCC2)=O)C2CCCCCC12 c1(C(=O)NCCC2(OC)CN(C(C(COC)(C)C)=O)C2)c(N)cccc1Cl N1(C(CC(C)SC)=O)CC2(CCCC(CNC(=O)CN3CCCCC3)O2)C1 C1(C(=O)NCC(CC=C)NS(=O)(=O)CC)(OC)CCN(C(=O)CN(C)C)CC1 N1(C(C2CCC(NC(CCOCC)=O)C2)=O)CCC(N2CCC(F)(F)CC2)CC1 C=CCC(C)C(=O)NCCNCCCN(CC(=O)NC)C(C)C C12(NC(=O)NC3(CCC(=O)OC)CCC3)CCC(OC(C)(C)C)C1C2 C1(C(=O)NCC2N(C(CC(C)O)=O)CC2)CCCCC1c1nc[nH]n1 c1(C(N(CC(C)NC(=O)C(C)n2ccnc2)CC)=O)ccc(C(C)(C)C)s1 Cc1cc(C(N2CCC(C)C2CNC(c2ccc(CO)nc2)=O)=O)sc1C CC(C)CCC(=O)N1CC(O)(CNC(=O)C(O)Cc2cnn(C)c2)C1 N1(C(COCC(=C)C)=O)CCN(C(=O)CNC(=O)CN(C)C)CC1C1CC1 C#CCCCC(C)C(=O)NC(C1CCN(C(=O)C(=O)Nc2ncc[nH]2)CC1)CO c1(CC)nc(-c2ccc(-c3nccn3CCO)s2)c2n1CCCC2 C1(C(=O)NC(CC=C)C)CCCCN1CCN(CC)C(=O)OC(C)(C)C N1(C(c2nc(C(C)=O)sc2)=O)CCC(NC(=O)C(C)CC2CCC2)C(C)(C)C1 CC1(C)CN(C(C2(C)CC2Br)=O)CC(CNC(c2ccn(C(F)F)n2)=O)O1 c1(C(N2C(CNC(c3c(C)ccs3)=O)COCC2)=O)ccc(Cl)c2cc[nH]c12 N1(C(C2=CCN(C)C2)=O)CCC2(CC2)CC1C(=O)NCCCc1cn[nH]c1 N1(C(C(CO)OC)=O)CC2(CCN(C(=O)Cc3csnn3)CC2)C1 CCCC(C)CC(=O)NCCCCCC(=O)NC(C(=O)OCC)C(C)O c1(CC(=O)NCC#CCNC(C(C)C2CC2)=O)ccn(-c2ccccc2)n1 CCCCC(F)C(=O)NCC1(C)CN(C(=O)CCn2ccccc2=O)CCO1 Cc1nc(NC2CCCCC2O)cc(N(C)Cc2ccccc2Br)n1 C(CC1=CCN(C(C2(C3CCCO3)CC2)=O)CC1)NC(C1CCN(C)C(=O)C1)=O CC(C)C(CC(=O)N1CCCC(NC(C2CSc3ccccc3O2)=O)C1)C(C)C CCCC(CC)C(=O)N1C2CCC1C(C(N1CC3CC3C3CC13)=O)C2 N(C1CCCc2ccoc21)C(C(CC(F)F)NC(Cc1c(C)cnn1C)=O)=O C1(CNC(c2n(CCC)ccc2)=O)CCCC2(CN(C(=O)C(F)(F)C3CC3)C2)O1 C=C(C)C(Br)C(=O)NCCCOCCN(C(=O)CC1CC2(CC2)C1)C C1(CNC(c2cc(C)[nH]c2)=O)CCC(C)CN1C(c1ncoc1C)=O C1(N(C(CC=C(C)C)=O)C)CN(C(=O)CN(C)C(=O)OC(C)(C)C)CC1(C)C N1(CC(=O)NC2CCCN(C(C3C4CC5C(C4)C35)=O)CC2F)CCc2ccccc21 c1(N2CCC(C)(CSC)C2)nc2c(c(=NCCCC3CCCCO3)[nH]1)COCC2 C=C1CCN(C(c2nccnc2C)=O)C(C(=O)NC(CCC)CCO)C1 CCCCC(CNC(C1(C)CCCC1C)=O)NC(=O)C1=NOCC1 c1(OC)ncnc(C(N2CCCC(NC(C3(C)CCN(C)C3=O)=O)C2)=O)c1F Cc1cc(C#N)ccc1NC(=O)C(C)Cc1ccc(OC(F)(F)F)cc1 c1(NC(N)=O)c(Br)cc(Cl)c(Br)c1Cl.C12CC(C1)NC2=O C(=O)(CCCn1ccnn1)N1C(CNC(=O)COCc2ccncc2)CC1 CC1C(=O)CCC1CC(N1CCCC1CNC(c1cncnc1)=O)=O C1(C(N(C)CCN(C)C)=O)CCCN(c2ccc(C(N)=O)cn2)C1 CC(C)CCCCCCN(C1CCOCC1C)C1CC1 C1(C(=O)NCC(CC(C)C)NC(CSCC=C)=O)CCCC2(CCCCC2)C1 CC1(C)c2ccccc2CN1CCOCc1ccccc1 C1(NC(c2cncc(SCC(=O)OCCn3cncn3)c2)=O)CC2CCC1CC2 C1(N(C(=O)C(C2(O)CCCC2)F)C)CCN(C(c2cnnc(O)c2)=O)CC1 c1(C(=O)NC(C(=O)NC(c2c[nH]ccc2=O)C)(C)CSC)ccc2c(c1)CC2 c1(C(=O)NCC(C)NC(=O)CSCCN(C)C)cccc2nnn(C)c12 C(=O)(C(C)(C)C(C)(C)C)NCC1CC(C)N(C(=O)Cn2cccn2)C1 C1(CC)CN(C(c2cc(-c3ccccc3)ns2)=O)CCC1NC(=O)CC1CC1 n1(C(=O)NC(CNC(Cc2ccc(OC)nc2Cl)=O)CO)ccc(=O)c(O)c1C CN1CC(C(=O)NCC2CCN2C(=O)Cc2ccc(-n3cccc3)cc2)NC1=O CC1CC(C(N2CC(C(C)NC(C3CC(O)C3)=O)C2)=O)CCS1 C(CC(C(=O)NCc1ncc(C)[nH]1)NC(=O)CC1CCCC2CC12)OCC N1(C(c2c(C)n[nH]c2)=O)CC2CCC(CO)(C2)C1.c12ccc(nc1)CNC2=O C1(NC(c2ccc(Cl)cc2)=O)CCCN(CCS(=O)(=O)NCCC2CCOC2)C1 CC(CCC(C)(C)C)C(=O)N1CCC(n2cc(CCOC(=N)O)nn2)C(O)C1 C1(NC(C(=O)NCc2c(C)n(C)nc2)=O)CC2(C1)CC21CCC1 N(C1CCCc2[nH]ccc21)C(c1cn(-c2ccc(C)cc2)nn1)=O C1(CC(=O)N(C(C(=O)OCC)C)C2CC2)CCCN1C(c1cnccn1)=O C1(OC)CCCCC1CC(=O)NC1CC1.C1(F)(C)CN(C(=O)Cn2nccn2)C1 C1(C2C(CNC(CCCC=C)=O)C2)CCC(C)(C)CN1C(=O)CC1CC1(C)C c1(C(=O)NC2CN(C(C(CC)(F)F)=O)CC(C)C2)cncc2ccc(F)cc12 C1(C(N2CCC(N(C(=O)CN(C3CCC3)C)CC)C2)=O)CCS(=O)(=O)C1 C1(C)(CNC(C=C(C)CNC(c2ccnn2C)=O)=O)CC2CCC1C2 C#CCC(O)C(=O)NC(CCC)C(=O)Nc1cnccc1CO Cc1ccc(C(=O)N(CCCN(C)C(C2CCCC3(CCC3)O2)=O)C)cc1C#N c1(CCCC(=O)NC2C(CNC(CC)=O)C2)nc2ccccc2[nH]1 C1(NC(Cc2cnc(C)[nH]2)=O)CC2CCC1CN(C(C1CCCO1)=O)C2 C1(CC(=O)NC(c2c[nH]ccc2=O)C)CCCN(C(C2(O)CCOC2)=O)C1 N1(C(COCCC)=O)CCN(C(=O)CCC2CCCN(C)C2)C(CC(C)(C)C)C1 C1(NC(c2cc(Cl)no2)=O)CC(C2CCN(C(=O)CN3C(=O)CNC3=O)C2)C1 c1(C(N2CCN(C(CC)=O)CC2C2CC2)=O)ccccc1P(=O)(CC)CC C1(N=c2nnn(C)[nH]2)(NC(c2cc(COC)c(OC)cc2)=O)CCCCC1 C1(C(C(F)(F)F)NC(C(CO)OC)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC1 c1(N2CCCCC(CNC(c3c(C)ccs3)=O)C2)ncnc2c1nnn2C(C)C N1(C(c2c(CC)cccc2)=O)CCC(NC(=O)CN2CCC(O)CC2)C(CC)C1 c1(C(N2CC(N(C(=O)CCn3cncn3)C)C(F)C2)=O)cnc2c(c1)CCCO2 c1(C(=O)NCC2(NC(C(n3cc(Cl)cn3)C)=O)CC2)ccc(O)c([N+](=O)[O-])c1 Cc1cc(F)sc1C(=O)NCC(=O)NC1(CO)CCC1 C(=O)(C1c2ccccc2C2CC1C2)N1C(C(=O)NCC(CCOC)OC)CCC1 Cc1cc(OC(F)F)c(C(N2CCC(CNC(=O)CC3CCCC34CC4)C2)=O)s1 C1(CNC(c2ccsc2CC2CC2)=O)CCCN(C(c2conc2C2CC2)=O)C1 C1(C(N2CCCC(C)C(NC(=O)CC3=CCOC3)C2)=O)CCc2nncn2CC1 n1(CC)cnc2nc(=NCc3nnc(C(C)C)s3)[nH]c(NCCCSC(F)(F)F)c12 C#CCC(CC(F)F)C(=O)NCCN(C)C(c1ncoc1-c1ccccc1C)=O C1(NC(c2onc(CC)n2)=O)CN(C(=O)C(O)COC)CC1SC C1(CC(=O)NC2CN(C(=O)COCCCF)C3CC23)CCCC2CC12 c1(CC)ccoc1C(=O)NC1CCC1NC(c1cc(COC)on1)=O Cc1cc(-c2nc(-c3ccco3)nn2-c2ccc(OC3CC3)cc2Cl)cc(O)n1 c1(OC)c(C(=O)NC2CC(NC(C3(CC4CCC4)CC3)=O)C2)ccc2c1CCC2 C=CC(C)(C)C(=O)NC(CNC(C1(c2cc[nH]n2)CC1)=O)CC(C)C N1(C(C(C)SC)=O)CCCOC(CNC(=O)Cc2ccc(NC(C)=O)cc2)C1 N1(C(CCCCC#C)=O)CC2CS(=O)(=O)CC2(CNC(=O)Cc2cncn2C)C1 n1(CC)cc(CC(N2CCC(NC(c3cnnn3C3CC3)=O)C2)=O)nn1 c1(C(N2C(CNC(c3c(C)nc(CCC)o3)=O)C(C)CC2)=O)ccc(F)nc1F N1(C(C(COC)NC(C)=O)=O)CCCC2(CCN(C(c3ccn(C(C)C)n3)=O)C2)C1 c1(C(N2CCC(NC(C3C(C)CC(C)O3)=O)CC2C)=O)cc(O)c(O)c(O)c1 C1(C(=O)Nc2cc(OCC)ncn2)CCCN(C(C2CCCC23CC3)=O)CC1 CC1CCn2ncc(C(N3CC(O)(CNC(c4ocnc4C4CC4)=O)C3)=O)c2C1 N1(C(CCCN(C(COC)=O)C)=O)CCC(CO)C12CCC2 CS(=O)(=O)C1(C(=O)OC(C2CC(N(C(=O)COC3CC=CC3)C)C2)=O)CCCC1 Cc1cccc(C(=O)N(C)CC2(O)CCN(C(C3CCCS3)=O)CC2)c1O N1(C(C2CC(CNC(C3(CC)COC3)=O)C2)=O)CCC2CCC12 Cn1ccc2cccc(CN3CCC(C)(NC(=O)CCN4CCOCC4)CC3)c12 c1(C(=O)NC(C)CCN(C(=O)CCc2nc(O)n[nH]2)C)ccccc1O C1(C(F)(F)F)(CNC(c2cc(C)sn2)=O)CC2CCC1CC2.C12CCN1C2=O C1(C(N(CCC(=O)NCCOCC#C)CC=C)=O)CCCOCC1 Cc1cc2cc(C(N3CCN(C(c4cc(Cl)n[nH]4)=O)CCC3C)=O)oc2cc1C O=C(C1=CC2(CN(C(=O)CNC=O)C2)OC1)NCc1ccnc(O)c1 c1(C(=O)NC2(C)C(C)CCC2)ccnc(N2CCN(C)CC2)c1I Cc1ccc(C=CC(N2CCN(C(c3csc(C)n3)=O)C(C)C2)=O)cc1 C(CCCCC(=O)N1CCC1C1CCC1)N(C(c1cn(C(C)C)nc1)=O)C C(=O)(CC(C)(C)n1cc(-c2cc(C(=O)O)cs2)nn1)NC(C)C C1(C)CCN(C(C2(C3CCCN3C(C)=O)CC2)=O)C1.C(C(C)(C)C)NC(COC)=O C1(NC(C2CN(C)C(=O)N2)=O)CN(C(=O)CC2CCC(C)(C)CC2)CC1(C)C N1(Cc2ccc(OC)cn2)CCC2CN(C(c3ccc(Br)c(C#N)c3)=O)CCC12 C1(CC=C)(C(=O)N(C(C)C(C)SC)C)CN(C(C23CSCC2C3)=O)C1 c1(C(N2CCC(CC=C)(NC(CCC=C)=O)CC2)=O)c[nH]c2ccncc2c1=O C=CCC(F)(F)C(=O)NC(CNC(=O)C(c1cccc(Cl)c1)O)CC(C)C CC1(C)CCC2(CC1)CC2C(N1CCOC(c2nc(C3CC3)no2)C1)=O CCC1=C(C(=O)NC2CCOC(CNC(C3CC3C)=O)C2)SCCO1 Cc1c(C(=O)NC2COCCN(C(=O)CNC(c3ccoc3)=O)C2)nn(C)c1N C(=O)(CC(C)(c1ccccc1)N(C)C)NCC1N(C(CCC2C(C)C2)=O)CC1 C1(NC(C2COC3(C2)CN(C(=O)NCCCl)C3)=O)CCc2ccccc2C1 C=CC1(C(=O)NC2CC(C)CN(C(c3ccc(N)cc3Cl)=O)C2)CCOCC1 c1(CNC(C2(C(C)C)N(C(CC(=O)OC)=O)CCC2)=O)cn(C)nc1C(N)=O C=CCC(C)(C)C(=O)N1CCC(CNC(c2ccc(CCC)[nH]2)=O)(OC)CC1 Cc1cc(C(=O)NCCCCC(C)NC(=O)CC(C)c2ccccc2)ccc1O C(C(=O)Nn1nnc(C)c1C)N(CCOC)C(C1CC(C)CC(=O)N1)=O C(=O)(CC(C)C(C)C(C)C)NCCNC(c1c(SCC)cc(Br)cc1)=O C1(NC(C(C)CN(C)C)=O)CC=C(C(=O)NCCc2cccc(O)n2)C1 c1(C(=O)NCC2N(C(c3ncc(N)nc3)=O)CCC2)cc2c(F)cccc2[nH]1 N1(C(C(C)SCC)=O)CC2C3CCC(C2C1)N(C(=O)C(=Cc1cccnc1)C)C3 N1(C(C2N(CC)CC2)=O)CC(C)(C)CC1CNC(=O)Cc1c(C)cccc1C N1(C(=O)Cc2cccc(F)c2)CCC(F)(C(=O)NCc2ccc(O)cc2)CC1 CC(C)(C(=O)NCc1nncs1)C1CCN(C(c2coc(O)n2)=O)C1 c1(OC)ncc(C)c(C(=O)NCC(C)CNC(C2CC(=O)N(C)C2)=O)c1Cl c1(CC(=O)NCCN(CC)CC)c[nH]c2cc(F)ccc12.c12cc(ncn1)N2 C1(C)(C(N(C(C2CCCO2)C)C)=O)CN(C(C23CSCC2C3)=O)C1 C12CCN(CC1)C2.CCCCCCOCC(=O)NC(C)C(C)NC(=O)CC(=O)OC c1(C(=O)NCc2c(C(NOCC=C(C)C)=O)cno2)c(Cl)cnn1C N1(CC(=O)N(C(C)C)CCN(C(=O)COCCF)C)CCCS1(=O)=O C1(C)(CNC(CC2C(OC)COCC2)=O)CCN(C(=O)C(F)=C(C)C)CC1 N1(C(C2CC(NC(C(CN(C)C)(C)C)=O)C23CCC3)=O)CCCC(C)(C)CC1 C1(CC=C)(NC(c2ccc(OC)cc2)=O)CCCN(C(=O)C(C)(C)OC(C)=O)C1 CN(C)S(=O)(=O)N1CCC(C(=O)NC2CCC2NC(c2csnn2)=O)CC1 Nc1cc2c(cc1C(=O)NCC1CN(C(=O)CNC=O)CC13CCC3)CCC2 N1(C(C(CC)C#N)=O)CCCC(O)(CCNC(c2cnc(-c3ccsc3)s2)=O)C1 CC(C)C(F)(CNC(=O)Cc1ccsc1)C(=O)NCC(=O)NC1CC1 C1(NC(c2cn(CCC(C)C)nn2)=O)C2CCN(C(C3CCCC3C)=O)C12 c1(OC)ncc(C(N2CCC(c3n[nH]c(C)n3)C2)C(=O)NC(C)C)cn1 C(C)(c1ccccc1Cl)=CC(=O)N(CCC(C)NC(C(C)(CO)OC)=O)C N12CC3CCCC3(C1)C2.C12(C)CCC(CC1)C2.C1(Cc2ccsc2)CCCCC1 c1(OC)[nH]c(=N)nc2sc(C(=O)NC(C)C(C)NC(=O)C=Cc3ccco3)cc12 c1(C(=O)NC(CN(C(c2n(CC)ncn2)=O)C)C)ccc(F)c2cnccc12 C#CC1(C)CCN(C(C2CC3CCC(C2)N3C(C2CCC(C3CC3)C2)=O)=O)CC1 c1(C(=O)NC(CC)CNC(C2(CF)COC2)=O)cscc1S(C)(=O)=O CC(C)CC(CN=c1[nH]nc(C2CCC2)s1)c1ccc(F)cc1 c1(NC(C2(CC)CN(c3cnn(C(C)C)c3C)C2)=O)cc(C)c(F)c(F)c1 c1(NC(C2N(c3cc(C)ncn3)CC(O)C2)=O)ncnc2ccsc12 N1(C(C=CC=CC=CC)=O)CCC(C(N)=O)C(NC(C2CCC2CC)=O)C1 c1(C(N2CCC(C)(NC(C(CC(C)C)O)=O)C2)=O)cc2c(C(F)F)nn(C)c2s1 c1(CN2CCCC(NC(=O)Cc3cncnc3)CC2)cc(F)c(F)cc1O C(=O)(C1CCCn2nccc21)NCC(C1CC1)NC(c1cncc(F)c1)=O c1(C(=O)NCCN(C(C23OCC(COC)(C2)C3)=O)C2CC2)cccc(N)c1O c1(CNC(c2n(CC(=C)C)nnn2)CCOCC)cncc(Br)c1C N1(C(CC2N(C)CCCC2)=O)CC2CCC1CN2C(=O)CS(N)(=O)=O CON(CCC(=O)NC(C)(C)C)C(=O)CC1CCN1C(=O)Cc1ccccn1 N1(C(C2C3(CN(C(COc4c(C(C)C)cccc4)=O)C3)C2)=O)CC2CC2C1C#N C(=O)(C1=CCc2ccccc21)NCC=CCNC(C1(OC)CCC(C)C1)=O C(=O)(C(N=[N+]=[N-])C(C)C)N1CC(F)CC(CNC(C(CC)(C)O)=O)C1 CC(CC(=O)NC1CC2C1CCN2C(c1nncs1)=O)C(F)F c1(CC)cnoc1C(=O)NC1CC(c2cn(CCC3CCOC3=O)nn2)C1 C(=O)(CC(C)C(C)C)N1CC(N2CCOCC2)(COCC(=O)OC)C1 N1(C(CN(C(C)=O)C)=O)CCC2(COC(CNC(c3ncc(Cl)cc3F)=O)C2)C1 N1(C(C(C2(C)CC2)NC(CCOCCC)=O)=O)CC(C2CC2(F)F)C1 C1(CNC(c2cc(SC)oc2)=O)(NC(c2cc(F)n(C)n2)=O)CCCCC1C C(CNC(=O)Cc1sccc1Cl)(CCNC(=O)CC(=O)NC1CC1)OC C(=O)(CC(C)C(=O)NCC(C)CC(=O)NC(c1ccnn1C)CC)OCC CCCC(CC)C(=O)NCC1(CC(N)=O)CCN(C(=O)CC2CC(SC)C2)CC1 C(=O)(C(F)C1=CCCCC1)NC1CC(NC(C(C)N(C)C)=O)C12CCC2 c1(C(N2C(C#C)CCCC2)C(=O)NCC)ccc2ncn(C)c2c1 c1(C(N(CCCCCNC(C(CC)CC)=O)C)=O)ccc(F)c(S(C)(=O)=O)c1 C1(C(C)C)CC(O)CN1C(c1ccc(F)s1)C(=O)NCc1ccc(Br)cc1 Cc1ccc(C(=O)NCCCCC(=O)N2CCC(c3nn[nH]n3)C2)cc1 c1(OC)ccc(CN(C)Cc2cc(Cl)c(Br)cn2)cc1Cc1ccccc1Cl CCC(C)CCC(=O)NC1CN(C(=O)Cc2cnn(C(C)C)c2)CC1C Nc1nccnc1C(=O)NCC(CC1CC1)C(=O)NC1(C)CC(OC(F)(F)F)C1 c1(OCCOC(C2N(Cc3c(OC)nccc3)CCCC2)=O)cc(C)ccc1Cl C12(c3c(-c4cn(C(COCC)C(=O)N(c5cscn5)CC)nn4)cn[nH]3)CCC(CC1)CC2 N1(C(C2C(COC)C2)=O)CCOCC1CCNC(c1n[nH]c(CO)c1Cl)=O C1(O)(CCNC(C2CSCC(=O)N2)=O)CCCN(C(C2(c3ccno3)CC2)=O)C1 Cc1nc(CC(=O)NCC23CC2CN(C(=O)CCc2cnc[nH]2)C3)c(C)s1 N1(C(c2n(CC)ccc2)=O)CCCC(NC(=O)CS(N)(=O)=O)C1C c1(C(=O)NCC#N)ccc(-c2c[nH]nc2-c2ccncc2)cn1 N1(C(c2c(C)nsc2)=O)CCCN(C(=O)C2=CCOCC2)CC1C c1(C(N2CC(CC=C)(NC(=O)C3=CCC(C)CC3)C2)=O)cnc2n1C(C)CCC2 C(=O)(C(F)CCC(C)C)N1CC(CC(=O)N(CC#C)C)OCC1 C1(NC(CC=CCC)=O)C(C)CN(C(c2cccc3cnsc23)=O)CC1C CCCC(CC)C(=O)N1CCC(N(C)C(c2cc(-c3ccccc3C)no2)=O)C1 c1(C(=O)NC2C(NC(c3c(OC(C)C)cccc3)=O)C2)cccc2c1C(=O)NC2 C(CCc1ccccc1)(C(=O)O)NC(CSc1cn(CC=C)nc1)=O c1(C(=O)NCC(CC)NC(=O)Cc2csnn2)cc(C(N)=O)cn1C N#Cc1cc(F)c(C(=O)NCC2OCCCO2)c(Br)c1 c1(C(N(C)CCN(C)C(C2CC=CCC2)=O)=O)cc(F)c(F)cc1F CCCC(O)CC(=O)N1CC(NC(C23CC(CC)(CO2)C3)=O)CCC1C CC(C)C(C(=O)N1CCC(C(=O)NCC2CNC(=O)C2)O1)NC(N)=O C1(OCC=C)CCN(C(c2nc(Cl)cs2)C(=O)NC(C)CC)C1 N1(C(c2c(CC)nn[nH]2)=O)CCC(CNC(C2CC(=C3CCC3)C2)=O)C(C)C1 C1(NC(CC(C)(C)OC)=O)CCC(O)CN(C(=O)CC2C(C)C2(F)F)C1 Cc1c(C(=O)NCC(C)(C)CC2CN(C(=O)CSC(C)C)C2)csc1Br c1(CCCC(=O)N(CCCNC(c2cn(C3CC3)cn2)=O)CC)ccc(C)cc1 N1(C(C2CCC(C#C)CC2)=O)CC2CCC1CN2C(=O)CC1CCCO1 c1(C(=O)NCC(=CC(=O)N(CC)CC2CCOC2)C)csnc1Cl N#Cc1c[nH]c2cc(C(N3CCC3C(N3CCn4nccc4C3)=O)=O)ccc12 c1(OC(C)C)ccc(F)cc1C(N1CC(NC(C2OCC2(C)C)=O)C(C)C1)=O N1(C(C2CCCC2)=O)CCC2(NC(=O)CNC(=O)C=CC=C(Cl)Cl)CC2C1.C1CC1 Cc1ccc(F)c2oc(C(=O)NCC(C)NC(c3cnncc3O)=O)cc12 c1(C(=O)NC2CN(C(C(CC)O)=O)CC2(C)C)c[nH]c2cc(F)c(F)cc12 c1(C2C(NC(C(N3CCC(C(C(=O)OCC)F)C3)=O)=O)C2)ccc(F)c(Cl)c1 C1(CCC)CC(NC(=O)NC2CC(=O)N(c3ccc(OC)cc3)C2)CCO1 C(C)(C(=O)NCC1CCN(C(c2ccno2)=O)C12CC2)(C(C)C)NC(C)=O N1(C(C2C(C)C2)=O)CC(CNC(c2cccc(-c3cscn3)c2)=O)C2(CC2)C1 N1(C(CN(C2CC2)CC)=O)CCC(C)CC1CNC(c1cc[nH]n1)=O c1(CC)ccc(C(N2CC(OCCC(=O)NCCCCSC)C2)=O)cc1 c1(OC)ccc(C)c(C(N2CCC(C)N(C(=O)C(O)CSC)CC2)=O)c1N C1(NC(Cc2cn(C)nc2)=O)C2CCCN(CCC3CCCCC3)C2C1(C)C c1(C(N(C)CCN(C)C(c2c(O)cccc2Cl)=O)=O)cncc(F)c1Cl c1(OC)ccc(CCC(=O)Nc2cccc(CC(C)CC(=O)O)c2)cc1 Cc1ccccc1C=CC(N1CC(CNC(c2[nH]nnc2C)=O)C2(CC2)C1)=O N1(C(COCCC#C)=O)CC2C(C1)C2(C)C(=O)OC Cc1c(C(N2CCOCC2CNC(=O)C=CC2CC2)=O)cc(C2CC2)n1C C12(CC(=O)NC3CCCCC3NC(c3ccnn3CCF)=O)COCC(C1)C2 C1(C)(CC(=O)NCC(C)C)CCN(C(=O)C=CC(=O)Nc2ncnn2C)C1 C1(NC(C=Cc2cncc(OC)c2)=O)CN(C(=O)CCC(C)C)CCC1(C)C CCCCN=C(NCC(=O)NC(C)C)NCC1(C)CCC(=O)N1 C#Cc1ccc(C(=O)NCc2ccnc(C(=O)NCC=C(C)C)c2)cc1C c1(N2CCC(C(C)NC(=O)CCN3CCCC3=O)C2)nc2ccc(Br)cc2o1 Cc1c(C(=O)NCC=CCNC(c2cc(N)c(Cl)cn2)=O)sc2ccc(F)cc12 Cc1cc(C(=O)NC(C)C(CO)NC(=O)CC2CC2)c(C)n1-c1ncccn1 C1(NC(COCC(C)C)=O)CN(C(c2ncsc2Br)=O)CC1C N1(C(C(C2CCC2)OCC)=O)CCC1CC(=O)N(CCOC)C(C)C Cc1cn2cc(C(N3CCC(c4cc(C)[nH]n4)C3)=O)cc2c(C)n1 C1(NC(c2ccc(CC)o2)=O)CC2CC1CN(C(=O)C(C)(C)CCSC)C2 C1(C(N(C2CCCN(C(C(CC)(F)F)=O)C2)CCO)=O)CCn2cncc2C1 c1(C(=O)NCC2CN(C(CCCSC)=O)CC2C)noc2cc(Br)ccc12 O(C1CCCc2ccccc21)CC(=O)NC1(CNC(C2C(=C)C2)=O)CCCC1 c1(OC)ncnc(NC(c2cnc(-c3ccnc(F)c3)cn2)=O)c1C CON1CCC(CC(=O)NCC2CC(C)N(C(=O)C(N3CCOC3=O)C)C2)CC1 N1(C(C2(C)ON=C(C)C2)=O)CCC2(CC1)CC(NC(C1CC1CN(C)C)=O)C2 O=C(CC1=CCCC1)NC(CCC1CC1)C(N1CCC(O)C(O)C1)=O C1(NC(N2C(c3c(CC)nco3)CC2)=O)CCCC(CC2(CC)CCOCC2)C1 c1(-c2c[nH]c(=NC)s2)ccc(CN(C)C)c(OC(F)(F)F)c1 C(=O)(C(C)(C)CCCF)N1CC(C)(C(=O)NC(C2CCCO2)C)C1 C1(CC(=O)NCCCC2(CNC(c3csnn3)=O)CCCC2)NC(=O)CNC1=O Cc1cc(C(=O)NC23CCCN(C(C4CCC5CC5C4)=O)CC2C3)cc(=O)n1C C1(NC(C(c2ccc(C)cc2)OC)=O)CN(C(=O)C=CC2CCOC2)CC2CC12 c1(-c2cn(CC3(CNC(C(CC)C4CCC4)=O)CC3)nn2)ccc(N)c(OCC)c1 N1(C(C(=O)NCCCC2(O)CC2)=O)CC2(C1)CN(C(C1CC1)=O)C2 CC(C)CCC(C(=O)N1CCC(C)(CCO)C1)NC(=O)C(=O)CC(C)C N1(CC(=O)NC2CN(C(C(C3CCC(=O)N3)C)=O)CC2C)C(=O)C(C)C(C)C1=O C(=O)(C1=CCCCCC1)NC(C(=O)N1CC(CCC)OCC1)CCCOC N1(C(C(COC)NC(C)=O)=O)CCC(C(=O)NCc2ccc(C)o2)CC1 C1(C(N(CCNC(Cc2cc(C)ns2)=O)C2CC2)=O)C(F)(F)C12CCC2 C1(CC=C)(NC(=O)CC(C)OC)CN(C(=O)CCCOCCOCC)C1 c1(CN(C(CC(C)n2ccnc2)=O)CC(C)C)ccc(F)cc1F.C1C(=O)O1 N1(C(c2nc(CC)sc2)=O)CCC(O)(C(C)CNC(c2cnc(Cl)[nH]2)=O)C1 c1(NC(C(N2CCS(=O)CC(C)C2)c2nc(C)[nH]n2)=O)ccc2c(c1)OCO2 N1(C(c2n(CC)nc(C(C)C)c2)=O)CC2(CCCN(c3cccc(SC)n3)C2)C1 c1(CC(=O)NCc2occ(C(N(C3CCC4CC34)C)=O)c2)cccc(F)c1 C(CCC(O)C(=O)NCC(C)CC1CCC1)NC(C1CCC(=C)CC1)=O C(CCC(C(=O)N1CC2CC1CN2C(C)C)NC(=O)CCc1cnn[nH]1)OC N1(C(CC2CC(CC)C2)=O)CCCCC1C1(NC(C2COCCO2)=O)CC1 c1(CNC(C2C(CC)C2)=O)ccc2c(c1)CCN(C(c1c(C)cnnc1O)=O)C2 CN1CC(C(=O)NCCC2CCCNCC2)c2ccccc2C1=O C1(CC)CN(C(C)=O)CCC1NC(c1conc1CSc1ccccc1)=O N1(C(=O)COCc2ccccc2)CC2CCCN(C(=O)CC3CCCOC3)C2C1 C=CCCCCCC(=O)N1CC2CCC2(CCNC(c2ccc(Cl)cc2)=O)C1 C12(C(=O)NC3CCN(C(=O)NC)C3)CC(CO1)N(C(C1(CC)CCNC1=O)=O)C2 C(=O)(CC1COC1=O)N1C(CCC(=O)NC(C)(C)C)CCC1.C(CF)OC Cc1onc(CO)c1C(=O)NCC=CCC(=O)NC1CC(n2ccnc2)C1 C1(NC(Cc2c(CC)noc2CC)=O)CC(C)N(C(c2cc(C)[nH]n2)=O)C1 N1(c2ccc(-c3ccc(C(=O)NC4CCOC4)s3)nn2)CCCC(O)(C2CC2)C1 C1(CNC(CCS(C)=O)=O)CC2CCC1N2C(C1(c2ccc(F)cc2)CC1)=O C1(C(=O)NCC2(O)CCN(C(C3(COC)CC3)=O)C2)CCCC(F)(F)C1 c1(C(=O)OC)cc(=NCCCCC(C)NC(=O)C2=COCCO2)[nH]c(Cl)n1 N1(C(CCCNC(S(C)(=O)=O)=O)=O)CC(F)CC1CC(=O)NCC1CCOC1 CC1(C)CC(NC(C2CC3(C2)CC(F)(F)C3)=O)CN(C(=O)C(CO)NC(N)=O)C1 Cn1ncc(C(=O)NC2CC2CNC(=O)CC2CC2(Cl)Cl)c1C#N c1(C(=O)NC23CC(NC(CCCCCC)=O)(C2)C3)ccn2c1CSCC2 C1(C(=O)NC(c2nnc(C)o2)C)CCN(C(c2cnc(Cl)n2C)=O)CC1O C1(S(N)(=O)=O)(CNC2C(Oc3cn(C)nc3)CN(C(c3ccco3)=O)C2)CCC1 C1(N(C(N(C2CCC(C#C)C2)C)=O)C)CCC2(CC1)CC2 CCC(CC)CCC(=O)NCCC(C)NC(c1ccc(F)c(F)c1N)=O C1(CC(=O)NC2(CC(=O)OC)CCC2)CCCN1C(c1cc(CSC)on1)=O C1(N(C(c2cc(Cl)on2)=O)CC)CCCN(C(=O)C(c2ccncc2C)C)CC1 c1(NCC(N2CCCC2c2cccc(Br)c2)=O)cccc2c1CNC2 C1(CC(=O)NCC(C)=CC(=O)OC)CC(C)N(C(c2ccc(C#N)[nH]2)=O)C1 c1(CC23CC(C(=O)NN4CC(N5CCC(O)CC5)C4)(C2)C3)ccc(Br)cc1F C1(C(=O)NCC2(C)CCCN2C(=O)CCCC2CCC2)CC2CCCCN2C1 C(=O)(C1=C2CCN=C2NC=C1)NC(C)(C)CNC(c1cn2ccsc2n1)=O Cc1cc(C(N2CC3CC2CN3C(=O)CCC(C)C)=O)cc(N)c1 C1(NC(C(C=C)O)=O)CCCN(C(=O)CNS(=O)(=O)CCC)C1 O=C1CC(C(=O)NC2CC(c3ccccc3)(CNC(=O)COC(F)(F)F)C2)CN1 C(CNC(C1CC1C)=O)(C(C)(C)C)NC(c1cnc(C)o1)=O C1(O)(CC#C)CC(C(=O)N(CC(C)C(=O)N(CCC(N)=O)CC)C)C1 Cc1cccc2c1OC(C(N1CC(C(C)NC(c3cc(C4CC4)[nH]n3)=O)C1)=O)C2 n1(C(CC(=O)NC(CN(C(c2ccc(CC)o2)=O)C)(C)C)C)nc(C)cc1C c1(C(N2CCN(C(CC(CC)SC)=O)C(CF)C2)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(C(F)=CC)=O)CC2CCCC2(NC(c2cc(=O)n(-c3ccccc3)[nH]2)=O)C1 N1(C(=O)CCc2cccnc2Cl)CCCCC(CNC(C2(CC3CC3)CC2)=O)C1 c1(C(N2C(C(C)NC(c3cscn3)=O)CCCC2)=O)nc2ccccc2cc1Cl C1(C(=O)NCCN(C(=O)C2=CC(O)CCC2)CC2CC2)CCCN2CCCCC12 c1(CCC(N2CC(CC=C)(NC(=O)C(O)C3CC3)C2)=O)c[nH]c2ccccc12 C1(CC)CN(C(=O)CCC#N)CCN1C(C1CC=CC1)=O CN=c1cc(C(=O)NC2(CCNC(C3(C4CCCO4)CCC3)=O)CC2)cc[nH]1 N1(C(c2cc(CC)on2)=O)CC(C2CC2)(C(=O)N(C2CCOC(C)C2)C)C1 c1(C(C)N(C)C(C2CC2c2cc[nH]n2)=O)cc2ccccc2[nH]1 CN1CCCCC(C(N2CC(CN(C(=O)CC3(C)CCOC3)C3CC3)C2)=O)C1 N1(C(CCC(C)OC)=O)CCCCC(NC(=O)CC2CCOC2)C1 C1(C(=O)Nc2cnc(Cl)c(Br)c2)COCCC12CN(C(C1CCCCN1)=O)C2 c1(C(C(N2CCC(NC(c3c(C)cns3)=O)C2)=O)O)ccc(OC(C)C)cc1 S(=O)(=O)(c1cccs1)NC(C(=O)NCC1CC(NC(C=C(C)C(C)(C)C)=O)C1)C C1(NC(=O)C=CI)CC(F)CN(C(c2sccc2C(F)F)=O)C1 N1(C(c2c(CNC(c3cn(C4CC4)nn3)=O)cco2)=O)CCCC(F)(CO)C1 c1(C(=O)Nn2cnc(NC(N(CCN(C)C)CC)=O)n2)ccccc1C(F)(F)F c1(C(=O)NCC2C(CNC(C(C)SC(C)C)=O)C2)cnn(CC(F)F)c1 CN1C(=O)CCC(C(=O)NC2CN(C(C3CSC3(C)C)=O)C2)C1c1nccn1C Cc1c(Cl)c(C(N2CCN(C3CCC(=O)NC3=O)CC2)=O)cn1C(C)C N1(C(C(CC)SC)=O)CCC2(CC1)OCCC2NC(c1ccnc(O)c1)=O c1(C(N2CC(NC(C34CCC(CC3)C4)=O)C3(CCC3)C2)=O)cccc2nccn12 C1(NC(C(C)NC(=O)OC)=O)CC2CCC1CC2NC(c1ccnc(C)c1C)=O N1(C(COCP(C)(C)=O)=O)CC2(CCC(NC(=O)C(O)C3CC3)CC2)C1 c1(C(N(C2CCN(C(c3nnn4c3CSCC4)=O)C2)C)=O)cc2ncccn2n1 C1(NC(c2cc(C)[nH]n2)=O)(CNC(=O)CNc2cccnc2)CCCCC1 c1(NC(c2c(C)nc(-c3ccc(SC)nc3C)s2)=O)nc2ccccc2nc1C C1(CC(=O)NCC2CN(C(c3cn(C(C)C)nc3)=O)CC2C)OCCCC1(C)C C(=O)(C(F)CCC(C)C)NCCN(C(c1c(C)nc(CC)o1)=O)C CCC(C)C(O)C(C)C(=O)N(CC(=O)NCCc1cc[nH]n1)CC1CC1 N(C1CN(C(=O)C2=COCCO2)Cc2ccccc21)C(c1ccnn1CCF)=O c1(C(=O)NCC2(NC(c3n(C=C)ncc3)=O)CCCCC2)cnn2c1CCC2 CC1CC(CNC(=O)CCCCN(C)C(C2CC(O)C2)=O)CC(C)O1 N1(C(C(COC)(C)O)=O)CC2CCC(NC(=O)C(C3CCCCCC3)O)CC2C1 C(=O)(CC(C)CC(F)(F)F)NCCC1CCCN(C(c2cc(C)c(C)o2)=O)C1 Cc1c(CC(=O)N(CCCO)C(C)C)ccc2c1CCC2 CC1CN(C(C2CCC(C(F)(F)F)O2)=O)CCC1NC(c1coc(Cl)n1)=O CC1(C)OCC(c2cn(CC(N3CCCC3c3nnc(C4CC4)o3)=O)nn2)C1O N1(C(c2c(C)[nH]nc2Br)=O)CC2(CCN2C(c2cc(F)n(C)n2)=O)C1 N1(C(CSc2nnc(C)n2C)=O)CCCCC(NC(=O)CN(C)C)C1 C1(NC(C2(CC(C)C)CCCO2)=O)CN(C(=O)CCSc2nccn2C)CC1C c1(C(=O)NC2C(NC(c3cnc(COC)s3)=O)CC2)c(C)ncc2ccccc12 C1(C(N(C)CCOCCC(=O)NC2CC(C)OC2=O)=O)C2CCC(F)(F)C12 C(=O)(C#CC(C)(C)C)NC1(C)CN(C(COCc2onc(CC)n2)=O)C1 c1(OCC(=O)NCC(CC)(C)NC(c2cnn(C)c2F)=O)ccc(C)cc1F Cc1c(NC(=O)NCCC(C)c2cn[nH]c2)ccn1CC1CC1 N1(C(CN(C)C2CC2)=O)CCOCC(NC(=O)CNC(C2CCC2)=O)C1 c1(C(N2C(C(=O)NCCc3ccc(Br)o3)CC2)=O)cccc(Cl)c1O N1(C(N(CC)CC)=O)CC2(C1)CN(C(=O)NC)C2 c1(C(=O)C(C)=O)cc(Cl)sc1NNCCCC1(NC(C(C)OCC=C)=O)CC1 Cc1cc2c(C(N3CCC(C4CCCN4C(=O)CN=S(C)(C)=O)C3)=O)cccc2[nH]1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCCC(F)(CNC(C2C=CCS2)=O)C1 C(C(O)CCCCC)NC(C1C(CC=C)CN(C(=O)CC(=O)OCC)C1)=O c1(SCC)cncc(C(=O)NC(C)C(C(C)C)NC(=O)C(C)(C)C2CCCC2)n1 N1(CCNC(=O)COc2ccc(F)c([N+](=O)[O-])c2)C(=O)c2ccc(Br)cc2C1=O c1(C(C)C(=O)NCCCCNC(C2CC2C(C)(F)F)=O)cccc(Br)n1 C1(CNC(c2c(CC)nns2)=O)CCCC2(CN(C(=O)C(=O)CC3CC3)C2)O1 c1(C(=O)NCC(C)N(C(CC(CC=C)(C)C)=O)C)cc2cccc(C)c2s1 N1(C(CC(C)(C)F)=O)CCCCC(CNC(c2ccc(Cl)cn2)=O)C1 N1(C(C(c2ccccc2)N(C)CC)=O)CC(O)(CNC(C2CCC(C)O2)=O)C1 c1(NC(C2(c3ccc(Cl)cc3)CC(C)C2)=O)cccc(C(C)(F)F)n1 c1(C(N2CCC(NC(C34COCC3C4)=O)C(O)C2)=O)cccc2sccc12 N1(C(C(CC)COC)=O)CC2CC1CN2C(C12CC(C1)C(C)O2)=O CCCCC(C)C(=O)NCC1CC2CCC1N2C(c1cc(C)n(C(F)F)n1)=O C1(NC(c2ccc(N(C)C)cn2)=O)C2COCC1CN(C(=O)CC1(O)CCC1)C2 c1(C(=O)NCC2C3N(C(CC4(OC)CC4)=O)C(CC3)C2)cccc2oncc12 N1(C(C2C(CC)C2)=O)CCCCC12CC(NC(c1ccnn1C1CC1(F)F)=O)C2 c1(CC)nc(C(=O)NCc2ccc(C(=O)NC(CC)C(N)=O)s2)co1 CC1CCN(C(C(=O)NCC2CCC2NC(c2nc(=O)n(C)[nH]2)=O)C(C)C)CC1 N1(C(C2(COC)CCOC2)=O)CCC(CC(C)NC(=O)CC=C(Cl)Cl)CC1 c1(-n2c(C)ncc2)ccc(NC(=O)C(=O)NCC(=O)N(c2ccccc2)C)cn1 N1(C(c2cn(CC=C)nc2)=O)CC2CC2(CNC(c2cc(C)c(C)s2)=O)C1 Cc1nc(F)ccc1-c1cccc(OCCN2CCCCC(N)C2)c1 Cc1cc(NC(C2CN(C(=O)CN3CC(C)(C)C3)CC23CC3)=O)c(C)cc1F c1(C(=O)OC)ccn2c1CN(C(=O)NC1CC3COCC13)CC2 N1(C(C2CC(C)=C(C)CC2)=O)CCC2C(C1)CN2C(=O)CC1CC2(CCC2)C1 N1(C(CN2C(c3onc(C)n3)CCC2)=O)CC(=O)NCC1C(C)C c1(C(=O)NC(CC(C)NC(CNC(=O)OC)=O)C)cc2ccccc2s1 N1(C(CCCCCN(C)C)=O)CC(NC(C2CC(C)(O)C2)=O)CC12CCOC2 Cn1cc([N+](=O)[O-])cc1C(=O)NC1CCC1NC(=O)CCC1CCCCO1 c1(C(N2C(C(=O)NC(C(C)F)C)CCCCC2)=O)ccc2[nH]nc(Cl)c2c1 N1(C(C2C(C)(Br)C2)=O)CC2=C(C1)CN(C(c1ccc(N)cc1Cl)=O)C2 Cc1cnc2n1CCC(C(=O)NCC1(NC(c3ccsc3Cl)=O)CCOC1)C2 Cc1cc(Cl)cc(C(N2CCOC(CNC(C3(C)CCOCC3)=O)C2)=O)c1N CC1(C)CC2(CN(Cc3cn(Cc4ccc(F)c(Cl)c4F)nn3)C2)C1 C1(C2CN(C(=O)C(F)CC3CCCC3)C2)(CC)CC1.O=CCCc1cnco1.C N1(C(CCC)=O)CCC2CC(NC(=O)C(C)(C)OCC(F)(F)F)CCC2C1 C1(CNC(CCOC)=O)(NC(c2cnn(CC(F)F)c2)=O)CC2CCC1C2 C(=O)(C1=CC2(CCN(C(CN3CCC(C)C3)=O)C2)C1)Nc1ccc(F)cc1F C1(NC(COCCC#C)=O)COCC1NC(c1ccccc1)=O N1(C(c2[nH]ccc2C2CC2)=O)CC2CC1CN2C(C12CCCC(C1)OC2)=O N1(C(c2c(C)cc(Cl)cc2)=O)CCC2C(C1)CN2C(=O)C(c1ccccc1F)C C1(CC(=O)N(c2ccn(CCC)n2)C)CC(C)(C)CN1C(c1cccn1C)=O Cc1nn(C)c2ncc(C(=O)N(CC(CO)(CO)NC(C3CC3F)=O)C)cc12 N12CCCC(C1)C2.n1(CC(=O)OCC)cc(C)nn1.C(CC(C)OOC)OCC(=O)NCC N1(C(c2cccc(C#C)c2)=O)CC2CCN(C(=O)C(C)CC(F)(F)F)C(C2)C1 C1(c2cn(CC(CNC(c3cc(C(F)F)on3)=O)OC)nn2)CCC(=O)CC1 N1(C(C(C)N(C(CC2CC(CC)C2)=O)CC)=O)CC2CCCC12 CC(O)C(C)(C)C(=O)NC1C=CC(CC(=O)NCC(C)(C)C(C)(C)O)C1 C1(CNC(c2ccn(CCNC(=O)CCCOC(F)F)c2)=O)NC(=O)NC1=O C1(C(N(C2CCOCC2)CCC)=O)CN(C(c2cc(Cl)cn2C)=O)CC(C)O1 N1(C(C(C)OCCN(C)C)=O)CCCCC1CNC(c1cnn(CC(F)F)n1)=O NC(Cc1cccc(F)c1)CC(=O)N1CCC(CC(=O)NC2COC2)C1 C1(CNC(=O)Nc2c(F)ccc(C#C)c2)CCC2(CC1)NC(=O)NC2=O CCCC(CCC)CC(=O)N(CC(C)(C)CNC(=O)C1=CC(C)(C)C1)CC C(=O)(CCCC(C)=O)N1C(C(=O)NC2CN(C)NC2=O)(CC)CCC1 C1(NC(Cn2c(C)ncc2)=O)CN(C(=O)Cc2cc(Cl)cc(Cl)c2)CC1N=[N+]=[N-] c1(CN2CCC(N(C)C)C2(C)C)cc2ccccn2c1.Cc1ccccc1N C(=O)(CCN(OC)C(=O)C1(CF)CCC1)N1C(C=C)CC1 c1(C(N2C(C(C)NC(CC3ON=C(C)C3)=O)CCC2)=O)ccc(F)c(C)c1N C1(NC(c2cc(C(N)=O)[nH]c2)=O)CCCCC1CNC(=O)CSCC(N)=O Cc1ccc(NC(=O)CN(C(=O)CCC(C)CN(C)C)C)c(Cl)c1 CC(CC(=O)NC(C)CC1CN(C(C2(CCOC)CCC2)=O)C1)C(F)F C1(c2n(CCOC)cnn2)CCCN(Cc2cnn(C(F)F)c2)C1 N1(C(=O)CSc2cn(CC3CCO3)nn2)CCC(Nc2ccccn2)CC1 C1(NC(C(CCC)(C)C)=O)CN(C(c2cc(C#N)ccc2O)=O)CC2(CC2)C1 C1(C(N2C(COC)CCC2)=O)(CO)CCN(C(c2cc(C3CC3)on2)=O)C1 c1(C(N2CC(C)C(CNC(c3ccc(Cl)cn3)=O)CC2)=O)cccc2ccoc12 c1(C(=O)NCC(C)(C2CCC2)NC(CSCCOC)=O)coc2c1C(=O)CCC2 Cc1c(NC2CCCN(CC(N)=O)C2)ncnc1N1CCCC(C#N)C1 c1(NC(C2(C3(O)CNC3)CC2)=O)cnc2ccc(Br)cn12 Nc1cccc(C(F)F)c1C(N1CC=CC(NC(C2CCCC3(CC3)C2)=O)C1)=O C1(C2CCCO2)(C(=O)NC2C(CNC(c3ccc4sncc4c3)=O)C2)CCCO1 C1(C(=O)NCC(C)CNC(c2ccoc2Cl)=O)CCOC2(CCCC2)C1 c1(C(=O)NCCN(C)C)cccc(Br)c1[N+](=O)[O-].C12CCCC13CCN(C3)C2=O c1(C(=O)NC(C2CCN(C(CSCCC)=O)C2)C)cnc(F)c(OC)c1 N1(C(=O)OC(C)(C)C)CCC(C)(C)C1NCC(O)CNc1c(Br)cnn1C N1(C(c2cccc(OCC(N)=O)c2)=O)CCC2(C1)CN(C(C1C3CCCC13)=O)C2 C#CCC(CC#C)C(=O)N(CC(CC)NC(c1cccc(C(F)(F)F)c1C)=O)C N1(C(=O)OC)CCC(O)C(C(=O)Nc2c(I)c(C)nn2C)C1 C1(C(C)NC(C2(CO)CCOC2)=O)CCN(C(C2CCC(=O)O2)=O)CC1 c1(C2(NCCCNC(C(C)n3cccn3)=O)CC2)csc([N+](=O)[O-])c1 c1(C(=O)NC2COCC2NC(C2CC23CCOCC3)=O)cc2ccccc2s1 N1(C(C)=O)CCCC1SC1CC(CCc2ccccc2)C1 c1(CC(N2CC(C)(c3cn(C4CC45CCOCC5)nn3)C2)=O)ncc(F)cc1F c1(C(N2CC(N(C(c3ccc(C)s3)=O)C)C3(C2)CC3)=O)ncc2cc(Cl)ccn12 C(=O)(C(C)(O)C(C)(O)C(=O)O)Nc1cn(C)c(=O)cc1 n1(CCC(=O)NCc2cn(CC3CCCNC3)nn2)ccc2cc(Cl)ccc12 C1(C(C)CCC(C)CC)C(=O)Nc2cccc(c2)CO1.C(CN(C)CC)OCC C[S+](C)CCC(O)C(=O)N1CCN(C(=O)CC(C)(C)C)CCC1C C(C(C(=O)N1CC(C(N)=O)CC(C)C1)C(C)C)NC(c1cc(CC)nn1C)=O CCC(C)CC(C(=O)N1CCC(C(=O)N(C)C)C1)NC(=O)Cc1cccnc1 C1(C(N2CC(N(C)C(c3csc(-c4ccoc4)n3)=O)C2)=O)CCCCC1(F)F Cc1nc(-c2cc[nH]n2)sc1CC(=O)NCCC1(C)CC1(F)F C1(C)(CNC(C2CCN(CC)CC2)=O)CN(C(=O)CCOC(C)C)CCO1 N1(C(c2cccc(C)c2)=O)CC2CCN(C(c3cc(C)c(C)cc3Cl)=O)CC2C1 c1(CN(CCOC)C(C2C(C)C2C)=O)cccc(OC(C)C)c1 C#CC1CN(C(=O)COC2CC=CC2)CCN1C(c1csc(O)n1)=O C(N=c1[nH]cnc(=N)[nH]1)C1CCCC(NC(C(C)C)=O)C1 N1(C(C2N(N=O)CCCC2)=O)CCCC2(NC(=O)CN3CCOCC3)CCCC12 C1(NC(N2C(C(N3CC(C)(CCO)C3)=O)COCC2)=O)Cc2ccccc2O1 Cn1c(C(F)(F)F)ccc1C(=O)NNC(F)F.C1(=O)CN1 CCS(=O)(=O)c1cccc(CC(=O)NC(CNC(C2CCO2)=O)C(C)(C)C)c1 C1(CNC(c2cn(-c3ccccc3)nn2)CO)CCCC12CC2 C1(NC(c2n(C)ccc2)=O)CN(C(c2cn(C)nc2Br)=O)C2(CCC2)C1 N1(C(C(CC)O)=O)CCC(C(=O)Nc2ccc(=O)n(C(C)C)c2)C(O)C1 c1(OC)ccc(C(=O)NC(C)CNC(C2(O)CC2(C)C)=O)c2cnccc12 C1(C(=O)NCCCC(C)=O)C2CC2CN1C(=O)CN1CCCC1=O c1(NC=O)ccc(C(=O)NC(CNC(=O)C(c2cccnc2)O)CO)cc1 CC1CCN(C(=O)CC(O)CN(C)C)CC1CNC(C1(C)COC(=O)OC1)=O C1(C(=O)NC2CC(C(=O)NCC3CC(C)C3)C2)CC2CCC1CC2 N1(C(CN2CCC(C)C2)=O)CCC(NC(=O)Cc2cn(C)nn2)C(O)C1 C1(=CC(=O)NCCC(=C)CNC(=O)CC(O)CC2CC2)CC2CCC(C1)N2C CC1CN(C(c2ccc(C(F)F)o2)=O)C(C)CN1C(=O)CN1CCS(=O)(=O)CC1 Cc1ccc2c(CC(N3CC4(CCN(C(c5cccnn5)=O)C4)C3)=O)c[nH]c2c1 CC(O)CC(=O)NC1(c2cc[nH]n2)CC1.c1(CN2C3CC(C3)C2=O)n[nH]c(=N)s1 C1(CNC(CSCCC)=O)CCN(C(c2ccccn2)=O)C12CCC2 c1(Cn2nc(CC)cc2C(F)(F)F)cnc2cc(C(N3CCC3CO)=O)ccn12 C1(F)(CNC(C(c2ccccc2)OC)=O)CCN(C(c2sc(C)cc2Cl)=O)C1 N1(C(=O)NC(c2nc(C)on2)C)CCCC2(CC(=O)N(C)C2)C1 N1(C(CCCC)=O)CCC(NC(=O)Cn2ccc(Br)n2)C(F)C1 c1(NCC)ccc([N+](=O)[O-])cc1C(=O)OC.C(CC)(CC(=O)OC)N c1(-c2nc(SCN3CC(c4nn[nH]n4)(OC)C3)no2)cc2c(F)cccc2s1 c1(C(N2CCN(Cc3cnc(O)c(Cl)c3)C3CC23)=O)cc(F)cc(F)c1Cl c1(NC(c2c(C)ccs2)C2CCC2)ccc(C2CCCN2N=O)cc1 C1(NC(C2(OC)CC2)=O)CCCCN(C(=O)CC2(O)CCCN(C)C2)C1 C1(C2CCN(C(c3cncc([N+](=O)[O-])c3)=O)C2)(NC(c2coc(Cl)c2)=O)CC1 c1(C(=O)NCc2cn(-c3ccc(F)cc3Cl)nn2)cnc(O)c2ccccc12 N1(C(C2C(C=C)CC2)=O)CC(F)(F)CC1CCNC(C1CC(O)C1)=O C(=O)(CCS(C)(=O)=O)NC(c1n(C)ncc1)C(=O)NC(c1cscn1)CO N1(C(C2C3CC(NC(c4c(CC)cc[nH]4)=O)C(C3)C2)=O)CCCC(N=[N+]=[N-])C1 N1(NC(C(=O)OCC)CCC2CCCCC2)c2ccccc2SC(C)C1C C=C(C)CC(C(=O)N(C(C)C(=O)NC1COC(C(F)F)C1)C)OC C1(N(C(c2cc(CNC(C(C)(C3CC3)OC)=O)no2)=O)C)COCC1(C)C CCC(C)CC(=O)NCCCN(C(C1CC2CC1C2)=O)Cc1ccccc1 c1(C(=O)NCC(C)(CC(C)C)NC(C2C(=C)C2)=O)cnc2cc(C)ccn12 C1(N(C(c2cc(COC)no2)=O)C)CCC(NC(=O)Cn2cnnn2)CC1 C1(C(=O)NCc2occc2C(=O)NCC2C=CCC2)C2COCC12 N12CC(C(C)(C)C1)C(=O)NCC1(CC1)C2=O.C1(C(=O)N)CC1C(F)(F)F.CO N1(C(C2C(CC)C2)=O)CCC(n2cc(C(=O)C(C)(C)C)nn2)C(C(F)(F)F)C1 C1(C(N(C2CC2)CC)=O)CC2CC2N1C(=O)Cc1cc(C)cs1 C(=O)(C(C)CN(C)C(C1(N(C)C)CCC1)=O)N(CCC)CCC N1(C(CC(C)(C)C)=O)CCC2(CCCC(C(=O)NCCN3CCC(O)C3)O2)CC1 c1(OC)cc(Cl)ccc1CN1CCC(CO)(NC(=O)C(C(C)C)OC)CC1 C1(CNC(=O)C=CBr)CC2(CCN(C(c3n[nH]c4c3COCC4)=O)CC2)CO1 c1(C(=O)NC(CN(C(c2c(OC)nc(Cl)cc2)=O)C)C)c(Cl)ccc(C)c1N Cc1cc(Cl)ncc1CC(=O)NC(C)(C)CCNC(=O)CCCn1c(O)nnc1O C12(CC(=O)OC)CCC1CN(C(C1C(Cl)(C(N3CCC(OC)C3C)=O)C1)=O)C2 CC1C(NC(=O)C=Cc2cccc(F)c2)CC2CCC1N2C(C1COC(=O)N1)=O C=CCC(C)(O)C(=O)NC1CCC(C)(CNC(=O)C(c2cccnc2F)(C)C)C1 N1(C(COC(CC)C)=O)CCN(C(=O)C(c2ccc(F)c(Cl)c2)C)CC1CO c1(C(=O)NCC2(C)CCCN(C(C3(CO)CC3)=O)C2)nc2ccccc2[nH]1 C1(N(C(C=C=C(C)C)=O)C)CN(C(c2ccc(=N)[nH]c2)=O)CCC1O CC1CC(NC(=O)Cc2cccc(F)c2)CN(C(=O)Cn2ccc(C3CC3)n2)C1 c1(NC(C2SCCCS2)=O)cnc2n1CCC2 C(CC(C(C)(C)C)NC(c1nccnc1N)=O)N(C(C(CC)F)=O)C c1(OC)ncnc(C)c1NC(=O)CC1(C)CCN(C(=O)Cc2ncoc2C)C1 C1(NC(c2nc(C(C)C)sc2)=O)CCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1O n1(CC2CCCN(C(CN(CC(C)(C)C)C)=O)C2)cnc2c1CCCC2.C1CO1 N1(C(c2n(CC)ncc2)=O)CCN(C(c2ccc(C#N)c(Cl)c2)=O)CC(CO)C1 C12(CNC(Cc3ccc(CCC)cc3)=O)CCC(CC1)N(C(=O)C(C)(C)O)C2 Cc1c(NC2CCN(Cc3cc[nH]n3)CC2)ncnc1NCC(C)CC(F)(F)F N1(C(CC2N(C)CCCC2)=O)CCCC(F)(CNC(c2cc(C(F)F)on2)=O)C1 N1(C(c2ccc(-c3cc[nH]n3)s2)=O)CCN(C(C2CCCCO2)=O)C(CF)C1 N1(C(CN(C(=O)OC)C)=O)Cc2ccc(CNC(c3sc(C)cc3C)=O)cc2C1 C1(C(=O)NC(C)(CNC(c2cc(Cl)on2)=O)C2CC2)CCC2(CCC2)O1 N1(C(c2ncncc2Cl)=O)CCCC1C1CCCN1C(c1cccc(=O)o1)=O Cn1nc(C(=O)NC(C2CCCCC2)CNC(C2CC2(F)Cl)=O)cc1C1CC1 CC1=NNC(=O)C1CC(=O)NC1(CC(=O)N(C2CCCC2C)C)CCC1 c1(CC(=O)NCC2CCCCN(C(CSCC(C)C)=O)C2)ccc2nn[nH]c2c1 C1(NC(c2c(O)cc(C)nn2)=O)C2CC3CN(C(c4cnn(CO)c4)=O)C1C3C2 N1(C(C(CC)C(=O)OCC)=O)CCCN(c2nnc(-c3ccccc3Br)o2)CC1C CCCCC(C(=O)NCC(C)C)N1C(C)CCC1(C)C C(C(O)CC(=O)NC1CCCN(C(c2ccc(CO)cn2)=O)C1)N(C1CC1)CC C(c1ccc(C)cc1C)=CC(N1CC(OC)(CNC(c2ncccn2)=O)C1)=O C1(OC)CCC2(C(=O)N(C)CC3C4CN(C(c5cn(C)cc5C)=O)CC34)CC12 C(=O)(C(C)(C)CC1CCOCC1)NCC1C(NC(CCOC(CC(C)C)C)=O)C1 Cn1[nH]c(C(N2CC(NC(c3sc(Cl)cc3Cl)=O)C(F)C2)=O)nc1=O C1(O)(C(=O)NCC(C2CCN(C(CC(=C)C)=O)CC2)(C)O)CCCC(C)(C)C1 c1(C(N2CC(C)(NC(c3sccc3C3CC3)=O)C2)=O)nccc2c[nH]nc12 Cc1nn(C)c2sc(C(=O)NCC3(O)CN(C(=O)CC(C)C(C)(C)C)C3)cc12 C1(C(=O)Nc2cc(C3CC3)ccc2Br)CCC2(CN(S(=O)(=O)C(F)(F)F)C2)O1 C(=O)(C(C)(C=C)CC)N1CCC(NC(C=Cc2cn(CC=C)nc2)=O)C1 N1(C(c2cc(CO)[nH]n2)=O)CCC(C(F)C(=O)NCC(C)(C)C2CCOC2)C1 Cc1cc(C)c(C(=O)NCC2(CNC(=O)CCCC(C)(C)C)CCCC2)c(O)n1 C1(CC)CN(C(=O)CCc2cc(Cl)no2)CCN1C(=O)C(C(C)CC)N(C)C c1(C(=O)NCCCn2cc(C(C)Sc3ccccc3Cl)nn2)cc(=O)n(C)cn1 N1(C(c2c(C)cc(F)cn2)=O)CC2CCN(C(c3sccc3C)=O)CC2C1 c1(OCC)ccc(C(N2CCOCC(NC(=O)CC3=CCCC3)C2)=O)cc1OC N1(C(=O)NC)CCC(C(N2CC(C)(NC(c3cc(C(N)=O)cs3)=O)C2)=O)C1 c1(C(C)=O)cc(C(=O)N(CCCCCNC(C23CC(C)C2C3)=O)C)oc1C C(CC(C)CCNC(C1CCCS1)=O)NC(CN(CC)CC)=O c1(CC(=O)NCC(CO)NC(C(C)OC)=O)nnc(S)n1C N(C(=S)N1CC(CO)OC(C)C1)C(c1ccccc1)C C1(NC(C(C=C)c2ccccc2)=O)(CNC(C2CCC2C(N)=O)=O)CCOCC1 N1(c2n(C)nc(C)c2Br)CCC2(CCCC2C(=O)NCCN(C)CCN)C1 C1(C(=O)NC2OCCN(C)C2)N(C(C2CCC3(CC3)C2)=O)CCCC1(C)C C(=O)(C(O)CNC(=O)C(=O)NC1CC1)N(C(C=C)C)C c1(SCC(N2CC(CNC(C=CC(C)C)=O)C2)=O)cc(CN2CCCCC2)on1 C1(NC(c2cnc(CNC(Cc3cn(CC)nn3)=O)s2)=O)CCCCC1CC C1(C(=O)NCCNC(c2n(CC)cc(Cl)c2)=O)CCCC(=O)CC1 c1(OC)cncc(C(=O)NCC2COCC2NC(c2ccc(N)cn2)=O)c1C c1(C(=O)NCC(C2CC2)NC(c2c(CC)con2)=O)csc(C)c1N S(=O)(=O)(c1cc([N+](=O)[O-])cc([N+](=O)[O-])c1)N1CCN(S(CC)(=O)=O)CC1 C1(NC(CCOCCNC(c2c(CCC)nco2)=O)=O)CC(C)(OC)C1(C)C C12(CNC(CC(CN(C)C)O)=O)CC(CO1)N(C(=O)COCCCF)C2.CCCC c1(NC(C)=O)ccc(C(=O)NC2CC2CNC(=O)Cc2ncnn2C2CC2)cn1 C(=O)(CC(C)CC(=O)N1CC(CC(N2CC3(CCC(=O)N3)C2)=O)C(C)C1)OC c1(C(CNC(c2c(SC)ccs2)=O)NC(c2cncnc2)=O)ccccc1F c1(C(N2CCOCC2CC(c2ccccc2)O)=O)ccc2c(c1)CCO2 CCC(C(=O)NC1(C(=O)NC2(C)CC(N(C)C)C2)CC(O)C1)C(C)(C)CC c1(C(=O)OCC(C)CNC(=O)Nc2ccccc2)ccc(Cl)cc1-c1ccsc1 N1(C(=O)NCC(C(CC)C)CO)CCc2ccncc2C1C CC(C)C(CNC(=O)CC=Cc1ccccc1)C(=O)N1CCC(N(C)C)C(O)C1 C1(Cn2cc(C3C(C(=O)OC)C3)nn2)CCN(C(C2CC2(Br)Br)=O)CC1 N1(C(c2c(C)c[nH]c2)=O)CCCCC(CNC(c2c(C)n[nH]c2C)=O)C1 N1(C(C23CCC(OC)(CC2)C3)=O)CCCN(C(=O)C=CCn2cncn2)C(C)C1 C1(NC(C(C)NC(N)=O)=O)CN(C(c2nc3ccccc3[nH]2)=O)CC1C1CC1 C12(CC(=O)NCCCC(C)NC(=O)CCS(C)=O)CC3CC(C1)CC(F)(C3)C2 CC1CN(C(c2ccc([N+](=O)[O-])s2)=O)CCC1NC(C1(N(C)C)CCCCC1)=O C(=O)(CCCC(CC)CC)NC1C(NC(CC(CC=C)(C)C)=O)CCC1 C1(NC(=O)CCC2CCC2)CN(C(=O)CSCc2ccncc2)CCC12CCC2 C1(CC(=O)N(CCNC(c2c(CC)c[nH]n2)=O)C2CC2)CCOC1(C)C Cc1cc(C)c(S(=O)(=O)NCC23CC2CN(C(c2ccc(O)cc2)=O)C3)c(C)c1 c1(OCCC(=O)N(CCNC(=O)C(CC2CCC2)SC)CC)cc(C)ccc1C c1(NC(=O)NCc2ccc(-c3n(C)c(O)nn3)cc2)ccc(F)c(Br)c1 c1(C(N2C(CNC(CCOCC)=O)CC(F)(F)C2)=O)ccc(C#N)c(Cl)c1 N1(C(CNS(NC)(=O)=O)=O)CCC(NC(c2ccc(C)nc2OC)=O)C(F)C1 C(=O)(CC1=CCN(C(c2cnco2)=O)CC1)N1CCC(OC)CC1 c1(CC)c(C(=O)NCCC(C)NC(c2nn(C(F)F)cc2Cl)=O)cccc1F CCCCCCC(F)C(=O)N1CCC(CCNC(c2ccc(COC)s2)=O)CC1 Cc1ccc(C#N)cc1C(=O)Nc1cccc(Br)c1F c1(C(N2CC(NC(c3cnc(S)nc3)=O)C2)=O)cc(C2(O)COC2)ccc1O Cc1cnc(CN2CCN(C(C3CN(Cc4ccccc4)CCS3)=O)CC2)nc1 C1(C)(CNC(c2cc(CNC(Cn3ncc(C)c3)=O)sc2)=O)COCCO1 N1(C(c2n[nH]c(C)c2Cl)C(=O)NC(CC)C)CCOCC1(C)C N1(C(C(COC)O)=O)CC2CCCC(NC(C3CN4CCN3C(C)C4)=O)C2C1 N1(C(C(CC=C)C)=O)CC2(CCC2)CC1C(N1CC(S(N)(=O)=O)C1)=O S(=O)(=O)(c1ccc(I)cc1Br)NC(C(=O)OC)Cc1nccs1 CC1ON=C(C(=O)NCCOCCCNC(c2cccc(=O)n2C)=O)C1C N1(C(c2c(CC=C)cccc2)=O)CCN(C(c2cc(N)ccn2)=O)C(C)C1 c1(C(=O)NCC(CC)(C)NC(=O)C=Cc2ccoc2)nc(C(C)C)ncc1Cl CC1CN(C(=O)Cn2nnc(=O)[nH]2)CC1NC(=O)Cc1cc(Cl)sc1Cl C1(C)(C(N2CC(C)C(NC(C3(n4cncn4)CC3)=O)C2)=O)CCC2CC2C1 C(=O)(C(C(C)C)NS(N)(=O)=O)N(C(CNC(c1c(OCC)scc1)=O)C)C n1(CC)nc(C(=O)N(C2CCC(NC(=O)C(=O)NCC(F)(F)F)C2)C)cc1C N1(C(C2(C#C)CC2)=O)CCC2(CC1)CC(C)N(C(=O)Cc1cc(F)cc(F)c1)C2 N1(C(C2(C(C)(F)F)CC2)=O)CC2CCCC(N(C)C)C2C1.c12cc[nH]c1C(=O)NC2 c1(OC)ccc(C(F)F)cc1C(=O)NC1CN(C(c2ccon2)=O)CCC1F C1(O)(CCNC(c2n(CC)ncc2Cl)=O)CCCN(C(=O)C(C)NC=O)C1 c1(C(=O)NCC2C(CNC(C(Br)=C(C)C)=O)CC2)cc2c(C)ccc(F)c2o1 N1(C(=O)CSC2CC2)CCCC2(NC(=O)CS(=O)(=O)Cc3cccs3)CCCC12 O=C(C1CCCn2c(Br)cnc21)N1CC(NC(C23CC(O)C2C3)=O)C1 c1(CN2CCCC(CCNC(c3nccc(C)c3F)=O)C2)cccc2occc12 C(=O)(C(C#N)C(C)(C)C)NC(C(=O)NCC1CCN(C(C)=O)C1)(C)CO c1(C(N(C(C(=O)N(C(CC)C)C)C2CC2)C)=O)csc(C)c1C c1(C(N2C(C)CC(NC(=O)C(C)(C)c3cnco3)C2)=O)ccc(C(N)=O)c(Cl)c1 C1(NC(CCN(CCC)C)=O)CC2CCC(C1)N2C(c1sccc1S(C)(=O)=O)=O C1(CNC(C(C(C)C)NC(C)=O)=O)COCCN(C(c2n[nH]c(C3CC3)n2)=O)C1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1)N1CCN(C(=O)NCc2nnc(CC)s2)CC1 C(=O)(C(CO)C(C)(C)C)NCC(C)CC(=O)NCCc1nncs1 C(C(=O)N1CCCCCO1)C1N(CC(=O)NC(CC)(C)C)CCCC1 CCCC(CNC(=O)CCOC(C)C)C(=O)N1CCOCCC1C C12(C(=O)NC(CC#C)CC#C)CCCC1CCN2C(C1CC(O)CN1C)=O c1(C(=O)NCC2(C(N(C(C)C)C)=O)CC2)ncn2ccccc12 N(C1CCOc2cc(F)ccc21)C(=O)NC1CC(C)(C)C(=O)O1.C1C(=O)N1 c1(CC)nc(C(=O)NCCC2CC(C(=O)NCCCN3CCC3)C2)c(C)o1 C1(C)(c2c(C(=O)NCCCN(C(C)=O)C)cccc2)NC(=O)NC1=O C(=O)(CC(C)C(C)(C)NC(=O)C1=COCC1)N1CCC2(C(C(C)C)C2)C1 Cn1cc(Cl)c(CC(N2CC3CC3(NC(C3CC3(F)F)=O)C2)=O)n1 c12ccc(cc1)CC(=O)NC2=O.C(C(F)(F)CC1CC1)NC(=O)OC(C)(C)C N1(C(CC(CC)C)=O)CCC(NC(C2CN(C)C2)=O)CC(C)(C)C1 N1(C(CCSCC(C)C)=O)CCC(NC(C2CCS2(=O)=O)=O)C(F)C1 N1(C(CCC)=O)CCC(CC2CC2)C1.c1(C(=O)N)ncoc1-c1ccccn1 C1(S(C)(=O)=O)(c2nc(-c3n[nH]c(C)c3Br)on2)CCC1 Cc1ccccc1-n1cnnc1O.C(=O)(C(CC1CC1)Cc1ccc(Cl)cc1)N c1(C(C)N(c2cncc(C(=O)NC3CC(N(C)C)C3)c2)C)ccc(C#N)c(F)c1 O=C(N=C1CCN(c2ccccc2)N1)c1ncccc1C(F)F C(=O)(CCCC(F)(F)F)NC1CC(C(N2CCC(C(C)C)CC2)=O)C12CCC2 C1(CNC(C2CC(CC)C2)=O)CN(C)CCN1C(c1cc(Cl)n[nH]1)=O c1(C(N2CC(NC(C(CC)(C)OC)=O)C(CO)CC2)=O)cn2cccnc2n1 Cc1cc(C(=O)NCCC2(C(=O)NC3(C)CC(N(C)C)C3)CC2)c[nH]1 S(=O)(=O)(c1ccc(F)c(C(=O)O)c1)N1CC2C(CNC(C3CC(=C)C3)=O)(C2)C1 N1(C(C(C2CCCOC2)OCC)=O)CCC(NC(=O)CCc2cnoc2)CC1 C1(C#N)(C(=O)NCCCCC(C)NC(=O)C(F)n2cccn2)CC2(CCC2)C1 N1(C(C2CCC3C(C)(C)C2C3)=O)CC2(CCSCC2)CC1CO C1(CC=C)(C(N2CCC(C)(CN(C)C)C2)=O)CCN(C(=O)C=Cc2ccco2)C1 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)NCC1CCN1C(=O)C(C)O C(=O)(C(F)(F)C(O)C1CC1)NC1CC(CNC(C2(C=C)CCCC2)=O)C1 Cc1cc(O)n2ncc(C(=O)NC3CCCN(C(=O)C(=O)NC4CC4)CC3)c2n1 N1(C(C(=O)NCC)=O)CCCC(C(=O)NC(C)C(C)(C)c2ccccc2)C1CC CC1(NC(=NCC2CC(=C(F)F)C2)NC(C2CC2)C2CC2)CCCOC1 C1(C(=O)NC2CC(C)(C(=O)NC3CC(C)CO3)C2)(COC)C=CCN1C(=O)OC N(C)(C1CS(=O)(=O)c2ccccc21)C(C1CCCC2CN(C(C)=O)CC21)=O C(=O)(C(CNC(c1cnsn1)=O)C(C)(C)C)N1CCC(OC)C1(C)C C(=O)(CC(CC1CC1)NC(=O)Cn1nnnc1CSc1cn(C2CC2)nn1)OC c1(C(=O)NC2CC(C)N(C(=O)CCSc3nnnn3C)C2)ccc(N)c(Cl)c1 Nc1cc(F)ccc1C(=O)NCCOCCNC(=O)C1=COCCO1 N1(C(c2c(C)coc2C)=O)CCC(CO)C(CNC(C2(C)CC=CCO2)=O)C1 c1(C(=O)Nc2ccc(CC)c(Cl)c2)ccc2ccc(O)nc2c1 N1(C(CN(C2CC2)CC)=O)CCC(C)CC1C(=O)NCC1CC1(C)C CCC1=C(C(=O)NC(CNC(=O)C2=CCCC2C)CCOC)CCCO1 C1(NC(c2ccc(SCC)nc2)=O)CCN(C(=O)Cc2cnns2)CC1O c1(C(=O)NCCCCN(C)C(C2CC2c2ccccc2)=O)cc(Br)cs1 c1(C2(C(=O)NCCCOCCCNC(C3CC3(Cl)Cl)=O)CC2)cccs1 N1(C(=O)N(C2C3CCC(=O)C32)C2CC2)Cc2cnn(-c3ccccc3)c2C1 N1(C(=O)NCC2CCCSC2)CCCC(O)(c2ccccc2)CC1 N1(C(CC(C(=O)OC)C)=O)CCC2(C1)CN(C(=O)CCC1CC1)C2 CCCCC(O)CCC(=O)N1CCCC1CN(c1ccc(Cl)cn1)C c1(NC=O)cc(CN2CC3CC3(C(=O)NCCCc3ccccc3)C2)ccn1 c1(-c2cn(C(C)C3CCc4ccccc43)nn2)ccc2ccncc2c1 C1(C(N2CCC(CN(C(Cn3c(C)ccn3)=O)C)C2)=O)CCn2c(O)nnc2C1 C1(CC(=O)N(CCN(C(C)C)C(c2cc(Br)cn2C)=O)C)CCC(C)(O)CC1 Cc1cccc(CNC(=O)CCC2CCCCN2C(c2nscc2C)=O)c1C c1(C(C)N(C2CCCN(S(CCC)(=O)=O)C2)C)ccc(F)cc1F C(CC(C)(C)CNC(C1CC(CN(C)C)C1)=O)NC(c1cc(CC)on1)=O N1(C(C)C)CCCC(C(=O)N(CC2CCCCC2)CC23CC(CCO2)C3)CC1 O=C(C1=CC2(CCOCC2)C1)NC1CCC(NC(=O)C(c2ccccc2)O)CC1 c1(N2CC(CNC(c3cccc(C(=O)OC)n3)=O)C2)nc2ccc(OC)nc2s1 C1(N(C(C(C)OC(C2(NC(=O)COCc3cccs3)CC2)=O)=O)CC)CCCCC1 Cc1cc(S(=O)(=O)N2CCSC2)ccc1-c1cnn(COC)c1 C(C(C(=O)N(C)C(C1CCCCC1)C)C(C)(C)C)NC(CC=C(C)C)=O c1(OC)ccc(C(=O)NC2CN(C(c3cnc4ccccn34)=O)C2)c(OC)c1Cl N1(c2c(C)c(N(S(=O)(=O)c3cccs3)C(C)C)ncn2)CCOC2(CCCOC2)C1 N1(C(COCC(=O)OC)=O)CCC(C)(CNC(c2sc(C)cc2Br)=O)C1 C(N=c1[nH]c(S(N)(=O)=O)cc2ccccc12)C1COCC(C)(C)O1 C1(C(=O)NCC(Cc2ccccc2)N(C)C)(OC)CCC(C)CC1 N1(C(C(C2CN(C(C(C)OCC=C)=O)C2)O)=O)CCOCC1COC c1(C(=O)NC(C2CCCCN2C(c2cc(CO)on2)=O)C)cc(C(F)F)ccn1 c1(N2CCN(C(c3c(Cl)ncc(C)c3)=O)C3(C2)CC3)ncnc2cc(F)ccc12 N1(C(C=CCN(CC)CC)=O)CCC(C(C)C(=O)NCC(C)(C)OC)CC1 c1(C(=O)NCCCN(CCCNC(C23CC(O)C2C3)=O)C)cc2cccnc2[nH]1 N1(C(C=CC)=O)C2CCC1C(F)C(NC(c1cc(C)cc(C)c1)=O)C2 CN1CCC(C(c2cn(CC(=O)NCC(c3ccccc3F)(C)C)nn2)=O)CC1 N1(C(c2c(OC)scc2)=O)CC2CCN(C(c3cc(C)ccc3C)=O)CC12 c1(C(c2nnnn2CCOCCOC)NCCOCC)c(Br)nnn1C.C Cc1nccc(Cl)c1C(N1CCN(CCN(C(=O)CCCCCF)C)CC1)=O CC1CC(C(=O)NC23CCN(CC2)C3)CN1C(=O)CCc1cncs1 Cc1nc(O)c(NC(=O)N(C2CCCC2)Cc2ccco2)cc1Br c1(OC)ccc(SCC(=O)N(C)CC2(O)CN(C(C3COCCC3C)=O)C2)cc1 CCCS(=O)(=O)CC(=O)NC(C)CC(C)NC(c1ccc(C2CC2)cc1F)=O c1(C(=O)NCC2(F)CC(CNC(c3ccc(CO)o3)=O)C2)ccccc1Cl CC(=O)C(C)CC(C)C(=O)N(C(CC(F)F)C(=O)NC1CC2CC1CC21CC1)C C1(C(N2C(COC)CN(C(=O)CC3(C#N)CC3)CC2)=O)Cc2ccccc2S1 Cc1cc[nH]c(=N)c1C(=O)N(CC(C)(C)CNC(C1CCCSC1)=O)C C1(C(=O)NC2(C(=O)NC(CC)CCO)CC2)CCC(=O)N(C)C1 C(=O)(C1=CC(C)(CC(=O)OC)C1)NC(C1CC(F)(F)C1)C#C C(CN=c1[nH]c(Cl)c(C#N)s1)C1N(C(CCCCCCC2C(C)CCNCC2)=O)CC1 C1(CCNC(C(C)(Cl)Cl)=O)NC(=O)OC1(C)C Cc1cc(C(=O)NC2CC3CN(c4cc(C5CC5)ncn4)CC23)cc2nn[nH]c12 CC1OC2CCC1(C(=O)N(CCCCNC(C1(CO)CCCO1)=O)C)C2 C1(C(=O)NC(COC)C(C)C)CC(C)(C)CCN1C(=O)Cc1ccccc1 c1(C(=O)NC2CCC2C(=O)NC2CC3CC4C(C3)C24)ccc2c(c1)CCC2 c1(CC)nn(C)c(C(=O)NC2CCN(C(=O)Cc3ccccc3C#N)C2)c1Br c1(OC)ccc(C(C)NC(c2nnnn2C2CCC2)CCC2CCCC2)c(C)n1 Cn1cc(C#N)cc1C(N1CCN(C(=O)C(F)F)CC1CCO)=O N1(C(=O)C=Cc2ccccc2Cl)CCC2C(C1)CN2C(=O)COC1CCCOC1 N1(C(C(C(CC)(C)C)O)=O)CCC2(CC1)CN(C(c1nc(C)c(C)[nH]1)=O)C2 C1(CC(N2CC(CCNC(C3C(C)(C(C)(C)C)C3)=O)C2)=O)CCC(=O)CC1 N1(C(CN(C2CC2)CC)=O)CC2CCCC2C1C(=O)NCC1CCCC(C)CC1 c1(C(N2CC(CNC(c3cc(C(CC)C)no3)=O)(OC)C2)=O)cnnc(CC)c1 [N-]=[N+]=Nc1ccc(C(=O)NC2COCCN(C(=O)Cn3nccn3)C2)cc1 N1(C(=O)C(C)(C)C)CC2(C1)CN(C(=O)C(C(C)C)Nc1[nH]cc(CC)n1)C2 c1(NC(C2CCN(C(C3(OCC)CCCC3)=O)C2)C)ncc(C(C)=O)cn1 c1(C(N2C(CNC(Cc3scc(C)c3)=O)CN(C)CC2)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(c2cccc(OCC#C)c2)=O)CCCCC12CN(C(C1OCCC1C)=O)C2 C(=O)(CC1=CCOCC1)NCCCN(C(=O)C(c1ccc(N(C)C)cc1)C)CC CC1CN(C(C2COCCN2C(c2cccc(O)c2)=O)=O)C(C)C1C c1(C(N2CCCCC(NC(CC(=C)C)=O)C2)=O)cnc2n1C(C)CCC2 CCCCCC(O)C(=O)NCC1(N(C)C(C)=O)CCN(C(=O)CCCSC)C1 Cc1nc(Cl)[nH]c(=NC2CCCN(C(C3(C4CCC4)CCC3)=O)C2)c1Cl C#Cc1cccc(CNC(=O)C(CCF)NC(=O)CCC2CCC(=O)C2)c1 N1(C(=O)OC(C)(C)C)CCCC(C)C1CCNC(c1cccc(N)c1I)=O N1(C(C2C(C(C)C)C2)=O)CC(OC2(CCC(=O)NOCCO)CCC2)C(C)(C)C1 C1(C(C)NC(CSCCOC)=O)CCCN(C(=O)Cc2cccc(Cl)c2)C1 c1(C(C2CCN(CC(=O)NC(c3cc(O)n[nH]3)=O)CC2)=O)cccc2cccnc12 C1(N(C(C(C)N(C(CCC(C)SC)=O)C)=O)C)CCCC(C)C1C C1(N(C(C(COC)(F)F)=O)C)CN(C(=O)COc2cccc(C)c2C)CC1(C)C c1(C(=O)NC2CCC(NC(c3n(CC)nnc3C)=O)C2)cccc(Cl)c1F C1(NC(c2c(CC)nc(C)o2)=O)CCC2CC1CN2C(c1ccncc1Cl)=O CC1=C(C(=O)N2CC(CNC(c3cn[nH]c3)=O)C(F)(F)C2)Cc2ccccc2O1 C1(Nc2nnc(C)c(C)n2)CCN(C(=O)Cc2cc(C3CC3)on2)CC1(C)C c1(NCc2ccc(N)cn2)ccc(S(=O)(=O)NCC2CC2(Br)Br)c(Br)c1 c1(C(N2C(COC)CN(C(c3cc(C)co3)=O)CC2)=O)cn2c(n1)CC(C)CC2 C1(CNC(C(COC)(F)F)=O)CC2CCC1N(C(=O)C=CCCC(C)C)C2 c1(C(=O)NCC(CN(C(C(CC#C)O)=O)C)O)c(F)ccc(Br)c1F N1(C(Cc2ccc(C(C)=O)o2)=O)CC(OC)CC1C(=O)NCCN1CCOCC1 C1(O)(CC(N2CC(CCNC(=O)CCCF)OCC2)=O)CCCCCC1 CP(C)(=O)c1ccc(C(=O)NC2CN(C(C3CC34CCOCC4)=O)C2)nc1 Cn1nnc2cncc(C(=O)NCCOCCCNC(C3(F)CCCC3)=O)c12 c1(CC)oc(C)cc1C(N1CC(O)(CNC(=O)CC2COC(=O)N2)C1)=O N1(C(C2(C)CCOC2)=O)CCC2(CCC2)C(NC(c2ccsc2)=O)C1 C(=O)(C#CC1CCCOC1)NC1(CC=C)CCCN(C(C2CCN(CC)C2)=O)C1 C(=O)(CC(F)(F)C(=O)O)N1CCCC(CNC(c2cn3cccnc3n2)=O)C1 CC1(NC(=O)C=Cc2ccoc2)CCN(C(c2cnc(N)c(CO)c2)=O)CC1 C#CCCCCCCC(=O)N1CCCC(CC(=O)NC(C)(CO)C(F)(F)F)CC1 C1(NC(c2cc(C)ns2)=O)CC2CCC1CN(C(=O)CCC(F)(F)F)C2 C=CCCCCCC(=O)NC1CCC(NC(=O)CCc2nc3ccccc3s2)C1 N1(C(C(CSC)OC)=O)CCCC(O)(CNC(c2ncnc(O)c2F)=O)C1 c1(C(=O)NCCN(CCOC)C(c2ccc(C#N)s2)=O)cnc2c(c1)CNC2=O c1(CC(=O)NC(c2cnn(C)c2)COC)ccc(C(C)(C)C)cc1 c1(C(=O)NC(CN(C(c2cc(C)ncc2C)=O)C)C)cc2c(C)ccc(C)c2[nH]1 c1(C(=O)NC2C(NC(CN(C(=O)OC)C)=O)CCC2)c(C)ccc2cccnc12 C1(C(=O)NC2(C)CC(NC(CC3(N(C)C)CC3)=O)C2)CC12CC(F)(F)C2 N1(C(C(Cc2cc[nH]n2)NC(CC2C(C)(C)CCO2)=O)=O)CC2C3CCC(C3)C12 CC(C)C(CN(C)C)C(=O)N1CC(CNC(=O)COC2(C)CCC2)(OC)C1 C1(CNC(C2CN(C(CCCNC(N)=O)=O)C2)=O)CCCC(F)(F)C1 c1(OC)ncc(NC(c2cn(CCNC(C3(C)CC(C)=NO3)=O)nn2)=O)cc1C C1(NC(c2c(C)onc2-c2ccccc2F)=O)CCCCN(C(=O)C2CC2)C1 n1(CCC(=O)NCC2CC(OC)CN2C(=O)CCC(C)(C)F)c(C)c(C)sc1=O c1(OC(C)(C)C)cc(OC(N2CC(CCC(=O)OC(C)(C)C)C2)=O)c(Cl)c(Cl)c1 c1(OC)cc(CC(=O)NC(c2sccc2Br)C)c(OC(C)C)c(Br)c1 CC1CCCCN1CCC(=O)NCCCN(C)C(c1ccc(=N)[nH]c1)=O C(=O)(CCC(C)(C)C)N(C(C)C(N1CCOCC1COC)=O)CCC c1(OC)cc(C#N)ccc1CN1CCC(F)(F)C(NC(C2(Br)CC2)=O)C1 N1(CNC(C2(C(C(C3CCC3)OCC)=O)CC2)=O)CC(COC)OC(C)(C)C1 c1(C(=O)NCC2(CNC(CC3CC(C)C3)=O)CC2)ccc(=O)n(C)c1 Cc1c(C(=O)NC2CN(C(C3CCCS3)=O)C2)ccc(Br)c1Cl N1(C(C(C)OCC#C)=O)CCC2C(C1)NC(=O)CN2C(c1cccc(CF)c1)=O N#Cc1ccc(CC(=O)NC2CCC(N(C(=O)C(=O)NCC(F)F)C)C2)c(F)c1 C1(C(=O)NCC2CCN2C(c2cc(F)c(F)cc2Cl)=O)CCCC2(CCOCC2)O1 C12(C(N(CC#C)CC)=O)CCCC1CCN2C(C1(OC(C)C)CCC1)=O CC(c1cnn(C)c1)=CC(N1CCC(C(C)NC(=O)C2CC2)CC1)=O S(=O)(=O)(c1cccnc1NCc1cc(C(F)(F)F)ccn1)NC(C(C)O)(C)C N1(C(C2(CC=C)CC2)=O)CCN(C(=O)CCC2CC2(F)F)C(C)C1 c1(OCC)ccc(S(=O)(=O)N2CCOCC2)cc1Nc1ncccc1F c1(CC(=O)NC2CC(F)CN(C(C3CC4(C3)CC43CC3)=O)C2)ccc(F)cc1Cl CC1CN(C(c2nn[nH]c2Cl)=O)CC1NC(=O)C(C1CC1)N(C)C C1(OC)CN(C(=O)Cc2ccns2)CC1NC(C1CC1F)=O CC1(CNC(C2(C)C=CCC2)=O)CCN(C(c2cc(Br)no2)=O)C1 N1(C(C2C(c3c(C)ccc(C)c3)C2)=O)CCCNC(=O)C1(C)C Cc1nc(C(=O)NCCC(O)CNC(C2CCCCO2)=O)c(C(F)(F)F)[nH]1 N1(C(C2C(CNC(=O)C=Cc3ccco3)CCC2)=O)CC=CC12CCOCC2 C1(C(=O)NC(CCC)CCO)CCCC(NC(C2(c3cc[nH]n3)CC2)=O)CC1 C(CN=[N+]=[N-])(C(=O)NCCN1CCCC1=C)NC(CC(=O)NCC#C)=O N1(C(CCCC=C)=O)CCN(C(=O)C2CCCn3nccc32)C2CCCC12 c1(C(=O)NC(CC=C)CNC(c2cc(OC)ncc2F)=O)c(C)ccc(Cl)c1O c1(C2C(O)CC2)nc(C(c2ccccc2)C2CC2)nn1C1CSC1 c1(C(=O)NC2(CC=C)CN(C(c3cnnn3C3CC3)=O)C2)ncsc1S(N)(=O)=O N1(CC)CC(C(=O)NC2CC(NC(=O)C(C(C)C)NC(=O)NC)C2)CC1=O c1(C(N(CCCCN(C(C2C(OC)CCC2)=O)C)C)=O)ccc2oc(O)nc2n1 C(CC(C(C)C)NC(=O)C=CCN1CCOCC1)NC(C(C)=C1CCCC1)=O c1(C(=O)NCC2C(NC(C3(COC)CC3(F)F)=O)COC2)cccc(N)c1F c1(NC(N2CCCC(NC(C)=O)C(F)C2)=O)n[nH]c2c1C(=O)NCC2 C(CC(N=c1nc2scnc2c(NCCC2CCc3ccccc32)[nH]1)C1CC1)SC C12(CNC(Cn3c(C)cc(C)n3)=O)CCC1CCN2C(C1CN(C)C1)=O c1(C(=O)NC(CNC(C(C)OCC=C)=O)CCOC)cc(F)c(OC)cc1F C1(NC(=O)Nc2cccc(C(=O)NC3CC3)c2)CCOC12CCS(=O)(=O)CC2 c1(Cc2onc(CN)n2)ccc(C(=O)Nc2ncccc2C(F)(F)F)cc1 c1(OCCC(=O)NC2CN(C(C(F)=C(C)C)=O)C(C)C2)cccc(Cl)c1Cl N#Cc1ccc(NC(c2nn(-c3ccncc3)c3c2CCC3)=O)cc1F C12(C(=O)NCCC=CC=C)CC1CCN2C(c1sccc1COC)=O CN=c1[nH]c(C(=O)NCC2CCC(NC(C3CCC34CCC4)=O)CC2)cs1 C1(C)(NC(C=C(CCC)C)=O)CC(NC(=O)C(c2ccccc2)OCC)C1 C(CCN=c1[nH]c(=NCC2CCC(F)(F)C2)[nH]c2c1SCC2)OCC=C C1(C(C)C)CCc2sc(C(=O)NC(c3cc(F)ccc3F)(C)CO)cc2C1 C1(C(C)NC(C=COCC)=O)CCN(C(=O)CN2CCOCC2=O)CC1 N1(C(C(=O)Nc2ccccc2)=O)CC(C2CCCN(C(c3cscc3F)=O)C2)C1 c1(CCC(=O)NC2CC(NC(C3CC34CC4(F)F)=O)C2)ccnc(Cl)c1 N1(C(C(C)OCC#C)=O)CCOC(CCNC(=O)CC(C)(C)C2CCCCC2)C1 CCC(CC)CC(=O)NC1CN(C(c2nc(C3CC3)ncc2Cl)=O)CC1(C)C C1(NC(c2c(CC)c[nH]c2)=O)CN(C(=O)CCP(C)(C)=O)CC2(CCC2)C1 N1(C(C(C)SCCCC)=O)CCC(N(C(=O)Cc2n[nH]c(=N)s2)CCC)CC1 N1(C(C(CCOC)C)=O)C(CNC(C2C3CCC2CC3)=O)CC2CCCC12 N1(C(C(C)Oc2cccnc2)=O)CC(NC(=O)C=Cc2cccs2)CC1(C)C C(CC(C)(C)CNC(c1ccc(OCCO)cc1)=O)NC(CCC=C)=O c1(N2CC(C)C(CNC(C3(C)CCC3)=O)CC2)nc(O)c2ccccc2n1 C1(CN(C(=O)CCCc2ccsc2)C)CCCN(C(=O)Cc2ccon2)C1 C(=O)(CCCS(N)(=O)=O)NCCC1N(C(C2OCCN(C)C2)=O)CCSC1 c1(NC(C(=O)NCCc2ncc(C)nc2)=O)ccc(Cl)cc1N(CC(C)(C)C)C N1(C(C2CCCC2)=O)CCCC(O)(CNC(C23CCCC2C3)=O)C1 Cc1ccc(C(C)C)cc1C(N1CC(NC(c2cc(CO)oc2C)=O)C(F)C1)=O c1(-c2n(-c3ccc(OC)cc3)nc(-c3ccn(C)n3)n2)cccc(Br)c1C C1(C(N(CC=C)CCNC(C23CC(F)C2C3)=O)=O)COC2(C(=O)OCC)CC1C2 C(=O)(CC(C)C(C)(C)NC(=O)C1CC1)NC(C)CCF C1(CNC(=O)CC2CC(F)(F)C2)CN(C(=O)C=Cc2cncc(F)c2)CCCO1 CC1=C(C(=O)N(C(C)CNC(c2cc(-c3cccnc3)on2)=O)C)CCCC1 C(=O)(C(F)(F)C1CC1)NCC(C1CC1)NC(c1nnnn1Cc1ccccc1)C N(C(=NCCCC(F)(F)C(F)(F)F)NCCF)CC1(C)CCN(C)C1 C(CC(=O)NCCc1nc(C)no1)(C(F)(F)F)NC(C1CCC(OC)C1)=O c1(C(=O)NC2C(C)CCN(C(C3(C#N)CC3)=O)C2)cc2cccc(Cl)c2o1 c1(OC)nccnc1C(=O)NC1CC(NC(C2CC(N3CCOCC3)C2)=O)C1.CCS C(CS(=O)(=O)CC(=O)N1CC(CNC(c2n[nH]cc2C)=O)N2CCC1C2)OC c1(CC)nnc(C)cc1C(=O)NCC1CCC(NC(C2COCC(C)(C)O2)=O)C1 C=C=C(C)CC(=O)NC(C)CNC(c1cn(-c2ncccn2)cn1)=O c1(CCC(=O)N(CCCCCNC(CNC(C(CC)C)=O)=O)C)ccc(O)cc1 N1(C(CCOC)=O)CCC(C(N2CCC(n3ccnc3)C2)=O)C(C)(C)C1 c1(CNC(C2CCN(C(CCc3ccc(C)s3)=O)C2)=O)ccc2nc(Cl)sc2c1 C1(NC(=O)C(=O)NCCC2CC2C(F)(F)F)CC2CC(Nc3ccccc3)C2C1 C(CCC(C)C(=O)N1CC2CC1(C(=O)NCC(c1ccccn1)O)C2)OC Cn1nnc2c1C(C(=O)N1CC3C(CNC(=O)CC4CCCC4O)C3C1)CCC2 CC1CC(CNC(C2CN(C)C(=O)N2)=O)CCN1C(C1CCCCC1(C)C)=O c1(NC(CC2(OC)CN(C(=O)CCOCCOC)C2)=O)cc(C)c(CO)cn1 N1(C(CCC2CCCN(C(C(C)n3cncn3)=O)C2)=O)CC2CCC1C(O)C2O C(C(CC(C)C)C(=O)N1CCS(=O)C(C)C1)NC(C1C(COC)CC1)=O C1(N(CC=CCCC=CCOC)CCN(C)C)CCCN(CC(F)F)C1 N1(C(CCc2c(C)n[nH]c2C)=O)CCC(NC(C2CCC3CC23)=O)C(O)C1 C(=O)(C(C)(C)C(=O)NCC(c1ccccc1)CNC(=O)C(C)(C)CO)OC N1(CC(C)NC)C(=O)CCN(CCC2CN(CCOC)CCO2)C1=O CCC(CCOC)C(=O)N1CC(O)CC1CNC(C1(c2cccs2)CCCCC1)=O C(C)(N=c1nn[nH]n1C)c1c(C2(NC(C3CCCC(F)(F)C3)C)CC2)cccc1 N1(C(C2CC(CCC)C2)=O)CCCC(N(C(=O)CSCc2cccnc2)CC)C1 CCCCCC(C)(CC)C(=O)NCC1CC1NC(=O)CCNC(=O)OC(C)(C)C N1(C(CC2CC(CC)C2)=O)CCn2ncc(CNC(c3c(C)csc3C)=O)c2C1 c1(CC)cc(C(=O)NC(C2CN(C(C3(C)C=CCC3)=O)C2)C)ncn1 C1(C(=O)NCc2ccc(-c3ccccc3)nc2)CCCC2(CCOC2)O1 C1(NC(C2(CN(C)C)CCCCC2)=O)CCN(C(=O)CCC2CCCC2)CC1O C(=O)(CC1=NNC(=O)C1)NCC1N(C)CCN(c2nnc(C)n2CCN(C)C)C1 c1(CO)c(NCC(=O)NC2CC2)cc(C)nc1O.C12(CCCC1)C(OCC)C(=O)O2 C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(C)CN(C(=O)C(N)=O)C(C)C1 CC#CCC(CO)NC(=O)C(C)(C)C1CCCN1C(=O)CCn1cccc1 CC1CCCC1CC(=O)NC(C)CCNC(c1cn(C2CC2)cn1)=O.N1(C)CCCC1 N1(C(C(C)NC(=O)NCC)=O)C2CC1CN(C(=O)CSC1CCOC1)C2 N1(CC(C)(C)OC(NC(C)C(=O)Nc2ccc(F)cc2)=O)C(=O)C2C=CCCN2C1=O N1(C(C)CNC(=O)NC(C)(C)C)CCc2ccccc21.N12CCOC(C1)C2=O n1(C(C)C)ncc(C(=O)NCC(C)CNC(=O)CC(C)F)c1N C(=O)(C(C)CC(C)C(C)=O)N1CCOCC(CC(=O)N(CC#C)CC2CC2)C1 c1(NCCCSC)ncnc(NCc2cc(F)ccc2F)c1C C12(NC(C=CCOC)=O)CCOCC1CN(C(c1cnc3ccnn3c1O)=O)C2 c1(C(=O)NC2CC(N(C(=O)CCC3CC3(C)C)C)C2)ccc(Cl)c(N)c1 N1(C(=O)C2=NOCC2)CCN2C(=O)C(NC(C3(Br)CC3)=O)CC2C1 N1(C(C2(c3c(C)occ3)CC2)=O)CCCC(NC(c2n[nH]cc2Cl)=O)CC1 c1(NC2CCN(C(c3c(CC)noc3C)=O)CC2C)ncnc2c(Br)nn(C)c12 c1(C(N2CCC(C(C)NC(c3c(C)cco3)=O)C2)=O)cnc2[nH]cc(C)c2c1 CCC(C(=O)NC(CC1CCC1)C(=O)NCC(F)CO)NC(N)=O c1(OC)cc2nn[nH]c2cc1C(=O)NCc1cccc(O)c1C CN1CC(CC(=O)N2C3CCCC2CN(C(C2CCCS2)=O)C3)c2ccccc21 C(=O)(C1Cc2ccccc21)NC1(CCNC(C=Cc2oc(Cl)c(C)c2C)=O)CC1 N1(C(C(C)=C2CCCC2)=O)CCC(NC(c2cc(C)cnn2)=O)CC1C C1(C(N2CC(CCCCNC(C3(C(F)(F)CC)CC3)=O)C2)=O)(CC)CC1(F)F c1(C(c2ccccc2Cl)OC)nc(-c2ccc(Cl)s2)nn1C1CSC1 CC1(CC(=O)NCC2CC2C(=O)NCC2=NOCC2)CCOC1 c1(C(=O)NCC2N(C(C3CCN(C(C)C)CC3)=O)CC2)c(F)ccnc1Cl c1(C(=O)NCCNC(C(COC)(C)O)=O)nn(C)c2c1CS(=O)(=O)CC2 C1(N(C(CCOCCOC)=O)CC2CC2)CCN(C(C2(C)CC2(C)C)=O)CC1 N1(C(C2=CCC(NC(COC(C)=O)=O)C2)=O)CCC(N(C)C)C(C)(C)C1 N1(CC(=O)N(CCCN(C(=O)CC2CSCCO2)C)C)CCCCCC1 Cn1c([N+](=O)[O-])cnc1C(=O)NCC1CC(O)(CNC(=O)CN2CCCC2)C1 N1(C(C2C3C(NC(CC4C(C)=NNC4=O)=O)C4C(C3)C42)=O)CCCC(C)(O)CC1 c1(C(=O)NCCC(C(=O)NCC(C)(O)CSC)OC)cc(C)c(C)cn1 C12(CNC(C(n3cc(-c4c(CC)cccc4)nn3)C)=O)COCC(COC1)O2 C1(C(=O)NC(C)CNC(c2ccoc2Br)=O)CCCCCS1(=O)=O c1(CCC(=O)NC(C)CNC(=O)C=CCN2CCCC2)cc(Cl)c2n[nH]cc2c1 c1(OC)cnc(C(=O)NCC2CC3CC2CN3C(c2cnn(C)n2)=O)c(OC)n1 C1(NC(c2c(C)ncn2C)=O)CN(C(=O)CCC=CC(C)C)CCC1CN(C)C Cc1c(C(N2CCC(N(C(=O)C(C)Oc3ccccc3)C)C2)=O)cccc1Cl C(=O)(C1=C(Cl)CCC1)NC1(CO)CN(C(c2ccc(N(C(C)C)C)cc2)=O)C1 C(=O)(C1CCSc2ccccc21)N1CCCC(N(C)C(C2CC3CC2C3)=O)C1 O=C(CCCCOC1CCCC1)NCC1(NC(C23C=CC(CC2)C3)=O)CC1 Cc1ccc(C)c(C(N2CCOCC2C(=O)Nc2cc(C3CCCCC3)no2)=O)c1 Cc1cc(F)c(C(N2CCC(C(C)NC(c3nccnc3C)=O)CC2)=O)c(Cl)c1 C1(CNC(COC)=O)CCC12CCN(C(=O)C(COC)CC(C)C)CC2 C1(Cc2c(OC(C)=O)ccs2)COCCC1C.c12cc[nH]c1C(=O)NOC2 C1(NC(C2N(C(C)=O)CSC2)=O)CN(C(c2nccnc2C)=O)CC1C c1(C(C(=O)NCCC(=O)NC2(NCC(F)(F)F)CCCC2)O)ccccc1F C1(C)(C(=O)NCC(CN(C(COCCCCC)=O)C)O)CC2CCC1O2 C(=O)(C(CC(C)C)C(C)C)N1C(C(=O)NCC2CCC2C)(COC)C=CC1 C1(CNC(c2sc(C)c(C)c2C)=O)CN(C(=O)CCCC#N)CCC12CCOC2 C1(CNC(C(C)NS(C)(=O)=O)=O)CN(C(c2cccc(C#N)n2)=O)CCC1(C)C C1(C(N2CC(NC(c3n(CC)cnn3)=O)C(C)(C)C2)=O)CCCCC12CCC2 c1(CC)ccc(C(N2CCC(C)C(NC(c3cnc(C4CC4)s3)=O)C2)=O)cc1F C12(NC(C(C)SC(F)(F)F)=O)CCN(C(=O)CCNC(=O)C(C)(C)C)CCC1C2 C1(C(C)C)CN(C(=O)CCC#N)CCN1C(c1cc2c(s1)CCC2)=O c1(SCC(=O)NC2C(OC)CN(C(=O)CC3CCCC3O)C2)cc(F)ccc1F N1(C(C(C)=C2CC2)=O)CCC2(CCCC2NC(C2(C(=O)N(C)C)CC2)=O)C1 C(C1=CCN(C(C2(C)CC2Br)=O)CC1)NC(c1n(COC)ncc1)=O N1(C(C(C)N2CCC2)=O)C2CCC1CN(C(=O)C(O)CC1CCOCC1)CC2 N1(C(C2(CC)COC2)=O)CCC(CCNC(c2ccnn(C)c2=O)=O)C(F)(F)C1 c1(C(N(CC(CC)NC(c2cc(OC)n[nH]2)=O)C)=O)nc2cccnc2s1 c1(CCC)ccc(S(=O)(=O)N(C)CC2CCCC2)cc1 C(N=c1[nH]nc(CC)o1)C1(O)CN(C(c2cnc(CCC)s2)=O)C1 C1(C(N(CCC(C)NC(c2csc(C)c2C)=O)C)=O)CN2CCCN1CC2 Cc1cccc(N(C)C(c2ccc(NC(C3CC(C)N(C(C)C)C3)=O)nc2)=O)n1 C(=O)(CC(C)C(=O)N1CCC(NC(=O)Cc2ccc(OC)c(F)c2)C1(C)C)OC O(NC(=O)C(C1(O)CCCCC1)NC(=O)CC1NC(=O)NC1=O)C(C)C S(=O)(=O)(c1ccc(C(N2CCCC2C2(O)CC2)=O)cc1)N(CCOC)CCO C(=O)(CC(C)(C(F)F)N(C)C)N1CC(F)(CNC(c2cnc(CC(C)C)[nH]2)=O)C1 CCCC(C)(C)CC(=O)N(C1CN(C(=O)C=Cc2cncc(C(F)(F)F)c2)C1)C CCCCCC1C(=O)N1.C(=O)(C(N)C(C)(C)C)N(CCOCCN)CC C1(C(=O)NCC2(NC(c3n[nH]c(C)c3C)=O)CCOCC2)CCC(C)NC1=O C(=O)(C(CNC(C1CN(C)CCO1)=O)(CC)CC)NCc1n(CCC)ncn1 N1(C(CC(CNC(CC2CC(SC)C2)=O)(C)C)=O)CCC(C2CCCC2)C1 c1(C(=O)NCC2COCCN(C(C(CC)SC)=O)C2)cc2c(cc1Cl)NCC2 C1(CNC(C2CCN(C(CC)=O)C2)=O)CCCCN1C(=O)Cc1nc(=N)[nH][nH]1 O=C(CCCCC(F)(F)F)NC1CN(C(=O)COC2CC(F)(F)C2)C1 C(=O)(C(C)(C)c1cnsc1)N(CCCNC(CN(C1CCSC1)C)=O)C1CC1 CCC(CCC(=O)NCC(=C1CN(C(c2ccc(O)nc2)=O)C1)F)OC C(=O)(CCCC(C)(C)C#N)NC1(CC)CN(C(C2CCCCNC2=O)=O)C1 c1(C(=O)NC2C=CCC(C(=O)NCC=C=C)C2)nc(C)ccc1C C(=O)(CCC(C)CC)N(C1CC(C(C(=O)NCc2c(COC)noc2)F)C1)C Cc1cc(NC(c2nnnn2C(C)(C)C)(C)CC2CCCO2)cc(CO)c1 c1(C(CC(=O)O)C)cccc2ccccc12.C(=O)(CCCCCF)OCCl N1(C(CCn2c(C)cc(C)n2)=O)CCCC(C)C1CNC(c1ccc(CO)o1)=O C(=O)(C(F)(F)CCC(C)=O)N(C)C(c1cc(C)n(CC)c1C)c1ccccc1 C1(CC(=O)NC2(CSC)CCC2)CN(C(c2cncc(OC(C)C)c2)=O)CCO1 CC(CCCNC(=O)CCC1CC1)NC(=O)C(c1ccccc1)C C1(NC(c2cc(C3CC3)ns2)=O)C2CCC1N(C(=O)Cc1ncncc1Cl)C2 CC(CC(F)F)C(=O)NCc1ncccc1CNC(c1cc(Cl)cn1C(C)C)=O C1(C(N2CC(C(C)OC)C2)=O)CC2CC1CN(C(=O)CN1CCCCCC1)C2 C1(C(=O)NCC2C(C(=O)NC)OCC2)CCN(CC)CCO1.C1(=O)C=CCO1 C12(C(=O)NC3C(CC)OCC3)CCCC1CN(C(=O)CCCCCNC(C)=O)C2 CCC(C)C(CC(=O)NC1(CO)CCSC1)NC(c1cncs1)=O C1(C(N2CCC(O)(C(C)NC(=O)CSCC(N)=O)C2)=O)CC2CCC1C21CC1 C(CCCOC)(C(=O)N1CC=CCC1)NC(C1CC(CCC)C1)=O C#Cc1ccccc1CC(=O)NCCCC(C)NC(=O)C(CCSC)NC=O CC(CCN=c1nc(N2CCOCC(C3CC3)C2)c2[nH]ccc2[nH]1)N1CCC1 C1(NC(CN(CCC)C)=O)CN(C(=O)C(C(C)C)NS(C)(=O)=O)CC(C)(C)C1 C1CC2(C1)CCOC2CNC1(c2nnnn2C2CC2)COC2(CCC2)C1 c1(OCC)ccc2c(CC(=O)NC)c[nH]c2c1.C(C)(CCSC)C1(CC(C)(C)C)CC1 C1(C)(NC(COCC(C)C)=O)CC(NC(=O)C=Cc2ncc[nH]2)C1 CC1(C)Cc2ccc(C(=O)N=c3ccn(Cc4ccncc4)[nH]3)cc2O1 c1(C(=O)NCCCC2(NC(c3cnc(C(F)F)s3)=O)CC2)cc(C(F)(F)F)n[nH]1 C(=O)(C(C)(CCC)CCC)N(C(CN(C(CC(C=C)(C)C)=O)C)C)C c1(C(=O)NC2C(C)N(C(=O)CC3CC4(CC4)CO3)CC2)ccn2cnnc2c1 c1(OC)ccc(C)cc1C(=O)NCCCC(C)NC(C1COC(=O)O1)=O O=C(CC1CCc2ccccc21)N1CCCCC1CNC(C1(O)CCOC1)=O c1(CC(=O)NCCCN(C(CC(=C)Br)=O)C(C)C)ccc(C)c(Cl)c1 C1(C(N2CCC(O)(CNC(C(CSC)C)=O)CC2)=O)CCc2cc(F)ccc2O1 Cc1ccc2c(N3CCCC3(C)C(=O)NCCC3CCCCN3C)ncnc2c1 CC(C)(C)CC(=O)NCCCNC(C1C2CCC(=O)C12)=O C1(NC(C(C)SC(C)C)=O)CN(C(=O)COC(F)F)CC2CC12 c1(C(=O)OC)c(C(N2CCC2(C)C2CCCC2)=O)sc2c1CCOC2 C1(CC(=O)NC23CC(NC(C(CCC)=CCC)=O)(C2)C3)CC2(CCC2)CO1 c1(CNC(c2n(CCC)nnn2)c2ccnn2C(C)CC)cccnc1Br C1(C(=O)NC2C(C(N(C3CCOC(C)(C)C3)CC)=O)CCC2)CC(=O)NC(=O)C1 c1(NC2CC2)ccc(NC(CN2C(CC)CCCC2)=O)cc1OC C1(C(=O)NCCC2(OC)CN(C(c3nccc(C)n3)=O)C2)CC(F)(F)CS1 N1(C(C2(C)C(C)OC(C)(C)O2)=O)CCOC2(C1)CN(C(c1ccc(=N)[nH]c1)=O)C2 N1(C(=O)CSC(F)F)CCC2CCC(C1)N2C(C1(CCCF)CC1)=O Cc1cc(NC(c2nc(C)c(C)[nH]2)=O)ccc1NC(c1csc(C(N)=O)c1)=O C(=O)(C(O)CC(F)(F)F)N1CCC(CCNC(c2cc(N)cc(O)c2)=O)C1 CCCCC(CC)CC(CC)NC1CCOCC1OCC1CC(SC)C1 CC1C(NC(c2ccc(N)cn2)=O)CCN1C(c1ccnc(-n2cncn2)c1)=O N(C(=NCN1CCCC1C)NCC1(COC)CCCC1)C(C)C.C1(CO)CCC(F)(F)C1 C1(C)(C(=O)NCCC(C(C)C)OC)CCCN(C(c2cc(C)cc(F)c2)=O)C1 C1(NC(C(C)OC2CCCCC2)=O)(CF)CCN(C(=O)CCNC(=O)C(C)(C)C)C1 N1(CC(C2CCCC2)CC)CCN(C)CC1.c1(C(=O)N)cnccn1 N1(C(C(C(=O)OCC)C(N2CCC(C(=O)OC)CC2)=O)=O)CCOCCC1CC C(CCCCC(=O)NC1CCCC1CNC(C12CCN(CC1)C2)=O)SC c1(N(CC(=O)NCC2(NC(=O)C(O)C3CC3)CCC2)C)cccc([N+](=O)[O-])c1 C(=O)(C1Cc2ccccc21)N(CC(C)NC(COCc1onc(C)n1)=O)C Cc1cccc(C(=O)NCCN(C)C(C2CCC3CC3CC2)=O)c1Cl CC1CCCC(CCNC(C2CCC(NC(=O)C3=COCC3)C2)=O)C1 C1(CC#C)(C(N2CC=CC(NC(c3ccc(Cl)s3)=O)C2)=O)CC=CCC1 C1(NC(c2csc(Cl)n2)=O)CC12CCN(C(c1cccc(CCO)c1)=O)CC2 C=C1CC(C(=O)N(CCCOCCNC(C2CC=CCO2)=O)C)(COC)C1 c1(CCC(=O)NC(c2cn(CC3(CO)CC3)nn2)C)ncc(C(C)(C)C)o1 N1(C(C(C(C)C)c2cnn(C)c2)=O)CCOC2(CCC(F)(F)CC2)C1 C1(O)(C(=O)NC2CC(NCc3cccc(OCC)c3)C2)CCOCC1CC N1(C(C(C)NC(N)=O)=O)CCC(CC(N2CCCC(C(C)(C)O)C2)=O)CC1 CCC(CCC(=O)NCCC1COCC1O)NC(C1(F)CCCCC1)=O c1(C2(C(N3CCC(NC(C(C)NC(=O)NC)=O)C3)=O)CC2)cc(Cl)ccc1F c1(CC)csc(C(=O)NCC(C2CCCC2)NC(=O)CCCNC(=O)COC)c1 c1(C(=O)NC2CC(NC(CN(CC)CC)=O)C2)ccc(Cl)c(C)c1O C12(CCCCC1)C(=O)NC2.C1(CC(=O)NC2(CC#C)CCC2)CCNC1=O c1(C(C)=O)cocc1C(=O)N(C(C)C(=O)NCCP(C)(C)=O)C Cc1nn(C2CCC2)cc1C(=O)NC1CCC1NC(=O)C(C)(C)c1ccn(C)n1 c1(C(=O)NC2(C)CCN(C(CN(C(=O)OC)C)=O)C2)cccc2c1CCC(=O)N2 C12(NC(C(C)Sc3ncccn3)=O)CCCC1N(C(=O)CCC(C)(C)O)CC2 C1(NC(CCOC(C)C)=O)CN(C(c2cccc(N)c2O)=O)C2(CCC2)C1 c1(C(C)C)ncc(C(=O)NC2CC2CNC(=O)C(C)CC2CCCCC2)cn1 O=C(C(Cc1cccc(Cl)c1)=NO)NC1CCC1NC(c1coc(Cl)n1)=O c1(CC)ccc(OCC(=O)NCC(C)(C2CC2)NC(C2CNC(=O)N2)=O)cc1 CC1(C(=O)NC2(C(N)=O)CCC2)CC=CCC1.C1CC(=O)N2CC(C2)OC1 C1(c2nnnn2C(C)C)(NOC(CCC)(C)C)CCC(C)(CC)CC1 C(=O)(CC(C)CC(C)(C)C)N(C(CC(N1C(C=C)COCC1)=O)CC)C C(CCC(=O)N(C(C)C(=O)NC(CO)C1CCC1)CC)=CC=C n1(CC)ncc(C(=O)N(C2CCN(C(=O)C(C)n3ccnn3)C2)C)c1Cl C1(CNC(c2cncnc2)=O)CC2(CO1)CN(C(C13CC1COC31CCC1)=O)C2 N1(C(CC(=O)OC)=O)CCC2(CC1)CC(NC(=O)CCc1cc(C)no1)CCO2 c1(C(N(CCCNC(C(n2c(C)ncc2)C)=O)C)=O)ccc(OCCF)cc1 C(=O)(C(CC(C)C)NC(C1CCCC1C1CC1)=O)NCC(=O)OCC c1(C(=O)NC2CC(N(C)C(c3nnn(C)c3N)=O)C2)ccc2nc(O)n(C)c2c1 C1(C(N2CCC(N(C(c3c(C)nc[nH]3)=O)CCO)C2)=O)CC2(C1)CC21CC1 Cc1c(Br)ccc(NCCCS(C)(=O)=O)c1[N+](=O)[O-] C1(NC(C2(C3CC3)CCN(Cc3cnsc3)C2)C)CC(C)CC(C)(C)C1 N1(C(COCCC)=O)CC(CNC(c2nccc(Cl)c2F)=O)CCC1C CC1(C(N2CCC2CO)=O)CCN(Cc2ccc(C(F)(F)F)cc2)CC1 Cc1cnc2c(C(=O)NC3CN(C(=O)C(C)C(C)(C)C)CC3O)cccc2n1 Cc1nc(C)c(CC(=O)NC2CCC(NC(c3ncncc3Cl)=O)C2)s1 C(C(C)C(=O)NC1(C(=O)NCc2ccc(Cl)o2)CSC1)SC C1(C(C)C)CN(Cc2cccnc2)CCN1C(c1ccnc(F)c1Cl)=O C(=O)(C1CCc2scnc21)NCCC1N(C(c2c(CC)nco2)=O)CCCC1C N1(C(CCNC(C)=O)=O)CCC(C2CCN(C(=O)CSc3cn[nH]c3)C2)CC1 CC1C(NC(=O)C(F)OC(F)(F)F)CCN1C(c1ccnc(O)c1)=O C1(F)(CNC(CC(CC)C2CCC2)=O)CCCN(C(C2(C)CCCN2C)=O)CC1 c1(CNC(C(=O)NCC(CSC)OC)=O)cn(C(C)C)nc1C C(=O)(CC(C)(C)CC(F)F)NCC1N(C(c2c(C)nsc2)=O)CC=C1 CC(C(=O)NC(C(=O)NCc1cscn1)C1(O)CCC1)NC=O N1(C(c2c(C)onc2Cl)=O)CCOCC(F)(CNC(c2cncn2C)=O)C1 C1(C(=O)NC(CCN(C(c2ccc(CCC)s2)=O)C)C)COCCN1CC C1(CN(C(C(C)(C)SC)=O)C)CN(C(C2COC(C)(C)C2)=O)CCO1 N1(C(c2nc(C(C)C)sc2)=O)CCC(C2CC2)(CNC(c2occc2Br)=O)C1 CCC(C)(C(=O)NCCC(C)NC(c1ccc(-c2ccncc2)o1)=O)OC C1(C(=O)NCCOC(F)F)CC2(CCN1C(C1C3CC4C(C3=O)C14)=O)CC2 C1(NC(c2ncn(C)c2)=O)CCOCC1NC(=O)CCc1cnco1 Cn1cc(C=CC(=O)NCC2CCCCC2NC(c2ccc(Cl)[nH]2)=O)cn1 C(=O)(C1CCCc2c[nH]nc21)N1CCN(C(C2COCCOC2)=O)CC(C)(C)C1 CC(CN=c1ccnc(NCc2c[nH]nc2C(C)(C)C)[nH]1)C(F)F N1(C(C(c2c(C)n[nH]c2C)C)=O)C2CCC(C2)C1CC(=O)NC(C)(C)CCF C(=O)(C1CCc2c[nH]nc21)NC1C(NC(c2nc(OC)c(F)cn2)=O)COC1 C(C)(CCC(=O)N1CCOC(CNC(=O)C(=Cc2cccnc2)F)C1)OCC C(C)(CCC(=O)N1CCSCC1C(C)NC(=O)CCCN(C)C(C)=O)SC C12(CCC(C(F)F)CC1)CN2.c1(C(=O)NCC)cc(C(F)(F)F)ccn1 c1(NC(C(=O)NCc2cnc(C(F)(F)F)s2)=O)ccc(S(=O)(=O)C(F)(F)F)cc1 N1(C(CC=CC)=O)CCC(C(N2CC(O)(C(F)(F)F)C2)=O)C(C)C1 C12(CNC(C3(C(=O)OCC)CC3)=O)CCCN1C2=O.C1(C)(CSC)CCCCC1.O(C)CCC c1(C(=O)NC2CCN(C(CCc3c(C)noc3C)=O)C2)ccc(S(C)(=O)=O)cn1 c1(C(=O)NC2C(O)CCN(C(c3n(CC)ccc3)=O)C2)nc2cccnc2s1 C12(C(=O)NCC3C=CC(NC(c4c(C)csc4)=O)C3)CC(C)(C1)OC21CCC1 Cc1nc(NC(c2cc(N)ccn2)=O)sc1CC(C)C CCCC(CCC)C(=O)NCC1OCCC1C(=O)NCCCC(O)CO C1(C(=O)NCCCCOc2ccc(CC)cc2)CC2CCCC1(N)C2 C(Cc1ccccc1)(C(=O)NCC(CO)NC(c1cnco1)=O)NC(CCC)=O C1(CNC(Cc2c(SC)cccc2)=O)CN(C(C2CC(F)(F)C2(C)C)=O)CCCO1 c1(C(=O)NCC2C(C(=O)Nc3cn(CCC#C)nc3)OCC2)nnc(O)nc1O C(=O)(CCCN=[N+]=[N-])NCC=CCNC(c1c(C)onc1Cl)=O c1(COC)cccc(C(=O)NC(C)CN(C(C2C(F)(F)C23CC3)=O)C2CC2)c1 N1(C(c2c(C)nsc2C)=O)CCC=C(CNC(C2CCCC(C)CC2)=O)C1 N1(C(CC2N(C)CCC2)=O)CCNC(C(=O)Nc2cnsc2)C1 c1(C2C(C(N(CCN(CC)CC)CC)=O)C2)cccc(C#N)c1.S(=O)(=O)(CCCC)N c1(CC)nc(N2CCC(N(C)C(c3cc(CC(C)C)on3)=O)C2)cc(C#N)n1 C(=O)(CS(=O)(=O)CC(F)(F)F)N(CCC(C(C)C)NC(=O)C(C)N(C)C)C C1(C(=O)NC2(C3CN(C(C4CSCCS4)=O)C3)CC2)CC12CCC(F)(F)CC2 c1(OCCC)ccc(C(=O)NCC(=O)Nc2c[nH]nc2SCC2CCCC2)cc1 c1(C(=O)NCC(C(=O)Nc2cc(C)c(Cl)cc2)O)cc2ccccc2[nH]1 N1(C(CC2N(C(C)C)CCC2)=O)CC2CC1CCN2C(c1ccc(F)c(Cl)c1)=O c1(C(=O)NCC2(F)CCN(C(C(C)(F)F)=O)C2)cc2cccnn2n1 O=C(CCC1CCOCC12CCC2)N1CC(O)C(O)CO1 Cc1cncc(-c2cn(CCCC(=O)N(C)C(c3nc[nH]n3)C)nn2)c1 c1(C(N2CCC(C)(CNC(C(C)=C3CC3)=O)C2)=O)cc2cccc(C)n2n1 CCCC(C(=O)OC)C(=O)N1CC2C(CNC(=O)CC34CCC(CC3)CC4)C2C1 C1(C(N2CCCC(C)(NC(CC=CC)=O)C2)=O)Cc2cc(C)ccc2S1(=O)=O C1(NC(C2ON=C(C)C2)=O)CCOCC1NC(=O)C=Cc1sccc1C C1(C)(CCC(N2CCC(OCC)C2)=O)CCCN1C(=O)CC(C)=C(C)C N1(C(c2cc(CNC(CCOC)=O)[nH]n2)=O)Cc2ccccc2C1 C1(CC(C)C)CCOCCN1Cc1cccc(C(F)F)c1F c1(C(Cc2cn(Cc3cc(C(=O)OC)n[nH]3)nn2)C)ccc(C(=O)OC)c(C)c1 N1(C(CC(C(=O)OC)(C)C)=O)CCC2CN(C(=O)Cc3cncn3C)CC2C1 N1(C(CC=CCC)=O)CCCC1CC(=O)N(c1cnn(-c2ccncc2)c1)CC c1(SCC(=O)NCC2CCC(NC(C34COCC3C4)=O)CC2)cccc(F)c1 N1(Cc2cnnc(C)c2C)CCC(=O)N(CCS(=O)CCCO)C1=O c1(C(=O)NC(C)CO)coc2c1CN(C(=O)C=CC1CCOCC1)C2 O=C(CCCn1cncn1)NCC(C1CC1)NC(C1CSC1)=O C(=O)(CC1=NN(C)C(=O)C1)NCC1(CO)CCN(C(c2c(C)nc(C)o2)=O)CC1 C1(CC)C(=O)NCCCN1C(C1C(C)CCN1C(=O)COC(C)=O)=O C1(NC(C(CC)CC)=O)CCCC12CCN(C(=O)CCC(=O)c1ccc(C)s1)C2 c1(C(=O)NCCCn2cc(-c3ncn(C(C)C)n3)nn2)ccnc(CO)c1 c1(CCN(C(C(CCC)OCC)=O)C)ccc(Cl)cc1Cl c1(C(=O)NC2(C(=O)NCC(C)OCCO)CSC2)cncc(F)c1 Cc1cc(C(=O)NC2(C(=O)NCC3=NOC(C)C3)CC(O)C2)sc1C N1(C(CC2(C)OCCO2)=O)CC2CCC(NC(C3CCCNC(=O)C3)=O)(C2)C1 c1(C(N2CC(CNC(=O)Cc3ccon3)C2)=O)cc(C2CCOCC2)[nH]n1 CC1=C(C(=O)N(CCC(c2cccs2)C2CC2)C)CC1.C1(CC(=O)NC)CC2(CC2)C1 C(=O)(C1=CCOCC1)N(C(CN(C(C=Cc1n(CC)ncc1)=O)C)C)C C1(CCNC(c2c(C)cccc2)=O)CN(C(=O)COCC(F)F)CCCO1 S(=O)(=O)(c1ccccc1F)N(c1cc(Nc2ncc(Br)nc2Br)ncn1)C N1(C(c2c(C)cncc2C)=O)CCC(NC(=O)C=C2CCC2)CC(C)(C)C1 c1(NC(CC2N(C(Cc3cnc(C)s3)=O)CCC2)=O)cn2cc(F)ccc2n1 c1(OC(C)C)ccccc1C(N1CCC(N(C)C(C23CCC2CC3)=O)C1)=O c1(C(N2C(CCNC(c3ccoc3C)=O)CC(OC)C2)=O)cncc(Cl)c1C C1(C(=O)NC2CC(C)(NC(=O)CC3CCC3)C2)COCC2(CCC2)O1 N1(C(C(C)NC(N)=O)=O)CCCCC12CN(C(C1(C)CCCNS1(=O)=O)=O)C2 C(=O)(CC(C)CC(C)(C)C)NC1CC(C)N(C(=O)CCC2CCCN2C)CC1 C1(NCC(c2cccc(Cl)c2)OC)CCN(C(=O)C=C(C)C(C)(C)C)CC1C N1(C(COc2cccc(C)c2)=O)CC2CC1CC2NC(c1c(F)cccc1F)=O c1(C(=O)NC2CN(C(CC(=O)NCC)=O)C(C)CC2)cc2cccc(C)c2nn1 C1(C(=O)NCC2N(C(Cc3ccn(C(C)C)n3)=O)CCC2C)CCS(=O)(=O)CC1 n1(C(C(=O)N(CC(C)CNC(C2CC2F)=O)C)C)cc(Br)c(O)nc1=O c1(C(=O)NC2C(CNC(C(CCCC)(C)F)=O)CCC2)ccc2c(c1)CCC=C2 O=S(=O)(CCCOC1(c2ccncc2)CCOCC1)NCc1ccccc1 C1(C(C)NC(=O)CN(CC(C)(C)C)C)CCCN1C(=O)CSC1CCCO1 N1(C(c2c[nH]c(CCO)c2)=O)CCOC(CCNC(C23CC(C2)C3)=O)C1 C1(NC(C2(CCC)CC2)=O)CCCCN(C(=O)C(CC)OC)C1 N1(C(CCCOC(C)C)=O)CCCCC1CCNC(c1nc(Cl)sc1Cl)=O C1(C(N2CC(CNC(c3cc(C)nc(C)c3)=O)C2)=O)CC2(CCCC2)CO1 C1(C(=O)NCC2CC(O)CN2C(C2(C3CCC3)CC2)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NC(C)CC2CN(C(c3coc(O)n3)=O)C2)cnc(N(C)C)cn1 c1(C(C(=O)OC)O)cccc(NS(=O)(=O)CCCC2CCOC2)c1 c1(Nc2cccc(NC(C)=O)c2OC)cc([N+](=O)[O-])ccc1N(C)C CC(C)C(C)(O)C(=O)N1CC2CCC2(CNC(=O)Cn2ccnn2)C1 N1(S(c2c(C(=O)OC)n[nH]c2)(=O)=O)CCc2cccc(C(=O)N(C)C3CC3)c2C1 c1(C(N2CC(CC(C)NC(C3CCC(F)(F)CO3)=O)C2)=O)cc(N)ccc1Cl C(=O)(C1CCc2c(Cl)cccc21)N1CC2(C(NC(=O)CSC(F)F)CC2)C1 Cc1nc2ccc(C(=O)NC(CC(N)=O)c3cn(CC4CCC4)nn3)cc2s1 C(=O)(C(C)(O)CC(F)F)N1CC(CNC(C(=O)N(C)C)=O)OCC1 C1(CNC(c2c(OCC)scc2)=O)CN(C(c2ncncc2N)=O)CCC1C Cn1nc(C(=O)NCC2CCCCN(C(C3COC(=O)C3)=O)C2)ccc1=O c1(C(N2C(CNC(c3c(SC(C)C)cccc3)=O)C=CC2)=O)ccc(O)c(Cl)n1 C1(COC)(NC(c2ccccc2O)=O)CCCN(C(=O)CCc2ccc(C)s2)C1 c1(C(=O)NCC(CC)NC(c2ccccc2OC)=O)cc(Cl)c(Cl)c(Cl)c1 c1(CNCC2CCCN(C(c3c(C#N)ccnc3)=O)C2)ccc(F)c(F)c1Cl c1(OC)nccc(CNC(=O)C(c2ccco2)NC(C2CC=CCC2)=O)n1 c1(C(=O)NC2CCN(C(c3scnc3C3CC3)=O)C2)c(F)cncc1Br Cc1ccc(F)c(CNS(=O)(=O)CCBr)c1.C12CC(F)CN1C2=O c1(OCC)cc(CNCCC(=O)NCCN(C)C(C)C)ccc1Br c1(C(=O)NCC(CCNC(c2cncc(C#N)c2)=O)O)cccc2cnccc12 C1(C(N2CCC(C(C(=O)OC)O)CC2)=O)CCCN(C(C)(C)C)C1=O c1(C(N2CC(NC(C3CCOC3)=O)CC(C)C2)=O)cccc2c1NC(=O)CC2 C(=O)(C1CCCc2cncn21)NCCN(CCC)C(c1ccnc(Br)c1)=O c1(C(N2C(C)(C(=O)OCC3CCN(CC)C3)CCCC2)=O)ccc(C#N)c(C)c1 N1(C(=O)CN2CCN(C(C3CC3Cl)=O)CC2)CCC2(CCC(O)C2)C1 C(C)(CC(=O)NC1CCN(C(C2CC2(C)C)=O)C1(C)C)(C(F)(F)F)N(C)C N1(C(CC2(CSC)CC2)=O)CCC(C)(CNC(=O)C(C)Cc2ccco2)C1 c1(C(CC(C)C)C)nnc(C2CCC2)n1-c1cccnc1.C1(C)CCO1 c1(C(=O)NCC(CCNC(Cn2c(=O)ccc(C)c2)=O)O)cccn2ccnc12 c1(C(N2CCCN(C(CC(C)C)=O)C(CO)C2)=O)cc2c(Cl)nccc2s1 N1(C(c2c(C)ocn2)=O)CC(C)(C)CC1C(N1CCC(F)(C(N)=O)C1)=O c1(COC(N2CCOC(CCC3CC3)C2)=O)cccc(F)c1 CC1CN(C(=O)CCOC2CC2)CCC1NC(=O)C(F)(F)C1CC1 Cc1ccc(CC(=O)NC2CC(O)(CNC(c3ccnnc3O)=O)C2)c(Cl)c1 C1(C)(CNC(CCC2CCCN(C(c3c(C)n(C)nc3)=O)C2)=O)CC2CCC1C2 C(CC(O)C(=O)NCCNC(C1CCCCN1C(C1CCCCCC1)=O)=O)SC CN1CC=C(CC(=O)N2CC(CN(C(=O)COc3ccccc3F)C3CC3)C2)CC1 c1(NCc2cccc(Oc3ccnc(CC)n3)c2)cc(CC)nc2ncnn12 C(=O)(C(C)C(C)C(C)(C)C)NCc1c(C)c(Cl)ccc1 c1(C(=O)OC)ccc2nc(NCC=CCNC(=O)COC3(C)CCC3)c(F)n2c1 c1(OC)ccc(F)cc1C(=O)NCC12CCC(NC(=O)CC3(CO)CC3)(CO1)C2 c1(NC2CC(OC)C(O)C2)ncc(S(=O)(=O)N2CCCC(OC)C2)cc1Cl N1(C(c2ccc(N)c(N)n2)=O)CCC2CN(C(c3cc(C(F)F)cs3)=O)CC12 C(=O)(C(CC=C)CC(C)C)N(C(C(=O)NC(C=C)C)C)C CCCCC(C)CCC(=O)NCC1CC(CC(N2CCC(C)(CCO)C2)=O)C1 CCCC(CCCNC(c1snnc1C(C)C)=O)NC(C1CCCC1(C)C)=O N1(C(C(CC2CCOCC2)NC(C(F)=C(C)C)=O)=O)CC(N(C)C)C(C)C1 Cc1ccc(C(O)C(=O)NCC(CNC(=O)CN2CCSCC2)CO)cc1 N(S(=O)(=O)N(C)CCSC)CC1(OCC)CCC1 C(C(C(=O)N1CC2(CNC(=O)O2)C1)C(C)(C)C)NC(CCOC(C)C)=O C1(C(=O)NCC2N(C(=O)CO)CCCC2)CCC2CCCC2C1 CC(C)C(C#N)C(=O)N1CC(NC(=O)CC(c2cccc(F)c2)O)C1 c1(CC)conc1CN(C)C(=O)NCC1CCC(O)C1 C1(C(N(CC(C)O)CCNC(CC2(CC)CC2)=O)=O)CN(C2CCC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC2C(N(C)C(C3CC(F)C3)=O)C2C1 O=C1CNC(=O)C(CC(N2CCN(C(C3CC=CCC3C(F)(F)F)=O)CC2)=O)N1 c1(NC(C2CC(SC)C2)=O)ccc(NC(c2c(C)nsc2Cl)=O)c(C)c1 Cc1cnsc1C(=O)N(C)CCN(c1ccccc1)C(c1ccncc1)=O C(=O)(C(O)CN1CCCC1)NC(CNC(C1(SCC)CC1)=O)C1CC1 c1(C(=O)NC(CNC(=O)C(C2CCCCC2)O)CO)cnn2cccc(Cl)c12 [N-]=[N+]=NC1COCC1NC(=O)CC1CCN(C(=O)C(=O)NCC(F)(F)C(F)(F)F)C1 c1(C(N2CC=C(CNC(C(C(C)(F)F)(C)C)=O)CC2)=O)ccc2c(c1)NC(=O)CS2 C1(CCC)CN(C(=O)CSC2CCOC2=O)CCN1C(c1ccn(C(F)F)n1)=O O(P(C)(=O)C1CN(C(=O)OC(C)(C)C)CC1NC(C1CC2CCC1CC2)C)CC c1(SC(C(CC)CC)c2ccccc2)ccc(Cl)c(OC(F)F)c1 N1(C(C2CCC(=C)CC2)=O)CCC2CN(C(C3CC(C(C)(C)C)=NO3)=O)CC12 c1(C(N2CC(C)C(NC(COC(C)=O)=O)C(C)C2)=O)c[nH]c2ccc(Br)cc12 c1(C(N(CCCNC(=O)C(F)C2CCCO2)CC)=O)csc(C(C)OC)n1 c1(CC(=O)N(CCCCNC2CCN(C(COC(C)=O)=O)C2)C)ccncc1Cl Cc1cn2c(n1)CC(C(N1CC3(CC3)CC1CNC(c1coc(Cl)n1)=O)=O)CC2 c1(-c2nc(C(C)=O)on2)cc(C=O)c([N+](=O)[O-])cc1F C1(NC(CCCCNC(C)=O)=O)CCC2CN(C(=O)C=C(C3CC3)C3CC3)CC12 c1(C(CNC(C2C(C)C2C)=O)NC(=O)C(F)(F)CC2CC2)ccc(F)cc1 c1(CCC)cc(C(=O)NCCCCN(C)C(C2CC3C=CC2C3)=O)n(C)n1 C1(=O)C(C(C)(C)C)N1.c1(CN2CC3C(C(=O)OCC)(C3)C2)ccc(Cl)cc1O C1(NC(C2CC(OC(F)(F)F)C2)=O)CCCN(C(c2csnn2)=O)C1 c1(C(=O)NC(CCC=C)C(=O)N2CCN(CC(C)O)CC2)nccc2[nH]ccc12 C1(CN(C(=O)C(C2CCN(C(=O)CCCN(C)C)C2)F)C)CCSCC1 c1(C(N2CCC(NC(c3c(CC)nn[nH]3)=O)C2)=O)cnc2c(c1)CCCC2 C(=O)(C(C(C)C)N1CCCS1(=O)=O)N1CC(NC(C=C(C)C)=O)(CO)C1 C(=O)(C(C)C(O)C(C)C)NC(CCC)CCC.C1=CC(=O)N2C1CCC2 c1(CC)ccc(C)cc1C(=O)NCC1(C)CCN(C(=O)CCNS(=O)(=O)CC)C1 C(C(C)(O)CC(=O)NCC(C)(C)CC(=O)NCC(c1cnc[nH]1)C)OC CCCCCCCCC(C(=O)Nc1cccc(Cl)c1C)N1CC(C)CC(C)C1 N1(C(C(c2ccc(Br)cc2)C)=O)CC(NC(c2ccnn2C)=O)CC2(CC2)C1 n1(CC(=O)NCCC=C=C)cc(NC(C2(CSCC)CC2)=O)nn1 C1(N(C(c2cnn(CC)c2C)=O)C)CCCN(C2CCCN(C)C2=O)CC1 C1(C(N(C)C)=O)CCN(C(=O)CCC2CCN(C(=O)CCC3CCCO3)C2)CC1 c1(C(C)(F)F)ccc(Br)cc1Cl.C1(NC(=O)C(=O)NC2CCC2)CCNC1 N1(C(C2(C)CSC2)=O)CC2CC2C1C(=O)NCCCN1CCCC1=O N1(C(CC2(NC(C)=O)CC2)=O)CC2(CCCC2)C1C(=O)NC1CNC(=O)OC1 Cc1ccc2c(c1)CN(C(C1(C)CCCN(C(C3CC(C)(C)C3)=O)C1)=O)CC2 N1(C(CC(=O)NCC2CC2)=O)CCC(C(N2CCC3CC3C2)=O)(CO)C1 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(Cc2ccc(C)o2)=O)CC1CCO N1(C(C(CCN(C)C)NC(c2cncc(OC)c2)=O)=O)CCC2(CC1)CC2 C1(C(=O)NCC2CN(C(=O)CC3CCCOC3)CCO2)CCC2CCCCN12 C1(COC)(NC(c2ccc[nH]2)=O)CCN(C(c2cnc(O)n2C)=O)CC1 C1(CC)CN(Cc2cc(Br)cnc2O)CCN1C(=O)CCC(C)=O C(CC(=O)NCC(C)NC(c1cnccc1C)=O)(C1=CCCC1)OCC c1(SCC(CNC(C2COC2)=O)NC(c2cn(CC)nn2)=O)cccc(F)c1 c1(CC)c(C(=O)NCC(c2ccccc2)NC(=O)CC(F)(F)F)cnn1CC C1(C(=O)OC)COCCN1C(=O)CCC(C)NC(=O)CC(C)OC N1(C(c2ccn(C(F)(F)F)n2)=O)CCC2(CCCN2C(c2ccc(CO)o2)=O)C1 N1(C(C)=O)CC(OCCN(C)C)C[Si](C)(C)C1.C(C(=O)O)(C=O)NCC Cc1cccc2cc(C(=O)NC3CCCC3c3cccc(Br)c3)nn12 C(CCC(C(=O)NC(C)CC)N1CCC(c2nc(CC)no2)CC1)OCC=C N1(C(C2CC(C#C)(O)C2)=O)CCC(C)C(CNC(C2CCCOC2C)=O)C1 C1(NC(CCc2cc(C)on2)=O)CCC(F)(CNC(=O)C(=O)NCC(F)(F)F)C1 c1(C(N(CCCCNC(C2CC2C(C)(C)O)=O)C)=O)cc(C(F)F)ccc1F C(CC(N)=O)(C(=O)NCCOCC1CCC(C(C)O)CC1)NC(CNC(CC)=O)=O C(CCCCC(=O)NCCc1cncs1)N(C(C1CC=C(C)CC1)=O)C N1(C(c2n[nH]c(=N)s2)=O)CCC2(CCC(NC(C34CC=CC(C3)OC4)=O)CC2)C1 C1(CCN(C)C(c2cccnc2S)=O)CCCCN1C(=O)C1=CCOC1 Fc1cc(N2CCCC(c3cc[nH]n3)C2)ccn1 c1(C(=O)NC2C(C)CN(C(=O)CC3CCCOC3)C2)ccccc1[N+](=O)[O-] Cc1cnn(C)c1CC(=O)NC(C)CC(C)NC(=O)Cc1cc[nH]c1 CCCCC(CCCC)NC(=O)C(CCCOC)NC(=O)CN1CC2CCC1C2 Cc1c(C(=O)N(C)CC=CC(N)=O)nnn1C(C)CI C(=O)(C1=CC2(CCOC2)C1)Nc1cccc(NCn2cc(CCCC(C)=O)nn2)c1 N1(C(C(CNC(C2(CC(C)=O)CC2)=O)N(C)C)=O)CCCC(O)C1 Cc1c(C(N2CC(F)(C(=O)Nc3cccc(CO)c3)C2)=O)cnn1C C(=O)(CCCCCS(N)(=O)=O)NCC1N(C(COCCC#C)=O)C2C(C1)C2 CCN=C(NCCOC1C(C)C1(F)F)NC1CC1c1ccccc1 C1(NC(C2(COC)CCC2)=O)CCN(C(=O)CNS(=O)(=O)C2CC2)C1 CC(C)CC(C)CNC(=O)C(C)(CO)NC(=O)CC1COCCOC1 C1(C(=O)NCC2C(CNC(COCc3n(C)ncc3)=O)C2)CCCC1(C)C c1(OC)ncc(NC(=O)CC2CCCN(C(=O)NC3CCCC3)C2)cn1 C1(CNC(C2(SC)CCC2)=O)CCCC1C(=O)NC(C1CCOC1)CO C1(CNC(C(COC)(C)O)=O)N(C(c2sc(C)cc2Cl)=O)CCC1(C)C C1(C(=O)NC2CC(NC(c3n(CC#C)ccc3)=O)C2)CC(c2ccncc2)=NO1 c1(OC)cccc(C(N2CCC(C)(NC(c3ocnc3C)=O)C2)=O)n1 C1(CC=C)(NC(=O)CCC2CC(NC(=O)CN(C)C(C)C)C2)CCC1 CCC(C)C(CC(=O)NC1CCCCC1(C)O)NC(c1c[nH]ccc1=O)=O C(=O)(C(C(C)(C)C)C1CCC1)NCCCCCCNC(C1(OC)CCCCC1)=O CC(C)S(=O)(=O)C(C)C(=O)N1CCOCC1CCNC(=O)CCc1cccs1 C(=O)(C1c2ccccc2CN1CC1CC1)N(CC=C)Cc1cc(Br)ccc1OC c1(OC)nccc(C(=O)NCC(CO)NC(=O)CNC(=O)CC(F)(F)F)c1F N1(CC(c2cccc(Sc3cnn(C)c3)c2)C)CC2(CF)CC1(C(=O)O)C2 c1(C(N(CC(C)CNC(=O)Cc2cnoc2)C)=O)ccnc(S)c1 C1(CC(=O)N(CCCCNC(=O)Cc2cncnc2)C)C=CS(=O)(=O)C1 CCC(COC)C(=O)N1CCC(OCC(=O)NCC2(O)CC=CC2)C1 N1(C(C2N(C)CSC2)=O)CC(F)(F)CC1(C)CNC(=O)C(C)(C)C(N)=O n1(CC)ncc(Cl)c1C(N1CC(CNC(=O)C(C)=CC(C)(C)C)C2CC12)=O C1(NC(c2c(Cl)ccc(OCC)n2)=O)CC2CCC(C1)N2C(c1cncnc1)=O O=C(CCCC#Cc1ccccc1)NC1CC1NC(C1CC12CCOC(=O)C2)=O C12(NCCNC(=O)NCC3(n4cnnn4)CCSCC3)CC1COC21CCC1 C(=O)(C(C)(C)n1ccnn1)N(C(C)C(=O)NCc1cnc(CC)s1)CCC c1(OC)ccc(C)nc1C(N1CCN(CC(C)(C)NC(C2CCCO2)=O)CC1)=O CC1=C(C(=O)NCC(C)(C(C)C)NC(C2SCCCS2)=O)C(=O)OC1(C)C N1(C(c2c(OCC=C)cccn2)=O)CC(C)N(C(=O)C(C)C2CCCC2)CC1C Cc1cc(C(=O)NCC2(C)CCCN2C(=O)C(C)(C)F)c2ncccc2c1 C#Cc1cccc(C(=O)NC(CCC2CCC2)C(=O)NCC(C2CCCC2)C)c1 c1(CC)cc(C(=O)NC2CC(CNC(C3CC4CCC3CC4)=O)C2)cn(C)c1=O N1(C(c2ccc(C)c(Cl)c2Cl)=O)CCC2CN(C(C3(C)CCCN3C)=O)CC2C1 Cc1cc(C(=O)NCC2(C)CCCN2c2nccn3nnnc23)cc(C)c1F N12CC(C3(CCCC3)C1)N(C(=O)C(CC)CCC)C(CCC)C(CC(CCC=C)C)C2=O CC1CCC(C)(C(N2CCC(CCNC(=O)C=C3CCN(C)C3)CC2)=O)C1 N1(C(C2OCCN(C(C(CC)N(C)C)=O)CC2)=O)C(C)CC2CCCC12 c1(CN(C)C(C2C(CNC(=O)CCc3ccnn3C)C2(C)C)=O)ncccn1 c1(OC)cc(C)c(C(=O)NC2CCOCC2NC(=O)CN2CCC(C)CC2)cn1 N1(C(C2(C)CC2(F)F)=O)CC2(CCC2NC(c2nncs2)=O)C1 C1(N(C(C2N(C(C)(C)C)CC2)=O)C)CCC(C(=O)NC2CC2)CC1 c1(NC(=O)NC(C)C(=O)NCC2(CCl)CCC2)ccccc1 N=c1[nH]c(=NCC2(CO)CCCCC2)[nH]c(=NCCC(O)C2CCC2)[nH]1 CCC(C)CCC(=O)N1CC=CC1(C)C(=O)N(C)CC1CCSC1 Cc1nc(C)c(-c2ccc(C(N3CCCC3(C)C(C)O)=O)o2)s1 C1(C(=O)NC(CC=C)CO)CC(C)(C)CN1C(c1ccc(F)s1)=O C1(C)(CNC(C2CCC(C)(CC)O2)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC1 CC1COC2(C1)CN(C(=O)C1=CCN(C(C3COCC3C(N)=O)=O)C1)C2 N1(C(c2cc(OCCN)c(CO)cc2)=O)CC2CCC(C1C(=O)O)N2 C1(COC)(CNC(c2cc(C)ns2)=O)CCCN1C(c1nc(O)sc1C)=O O=C1CN(C(C2CCC2CNC(C2C=CCCC2)=O)=O)CCN1CC1CC1 c1(N(CCCNC(C(C)SCC)=O)C)sc(Br)nc1Cl C1(CC(=O)NCCOCCN(C(=O)CC2CCC2)C)COCC2(CCC2)O1 Cc1nc(=N)[nH]cc1C(=O)NCC12CC1CN(C(c1c(O)nnc(C)c1C)=O)C2 c1(C(=O)NC(C(C)C)CCN(C)C(C2CCCS2)=O)ccc(N)c(Cl)c1 c1(CCC(=O)NC(CC)CNC(=O)C(CSC)OC)c(C)[nH]c2ccccc12 C(=O)(CCCC(C)(C)CC)NC(CC)CNC(=O)Cn1nnc(C)n1 CC(CO)(C(=O)N1CC(c2cc(O)no2)C1)NC(C1COC(=O)N1)=O c1(C(N2CCCC(NC(COC(C)=O)=O)CC2)=O)ccc(Cl)c2ccccc12 C(=O)(CC(F)(F)F)NCC(=O)NCCC1N(C(CCNC(N)=O)=O)CCC1.C(N)(=O)N N1(C(c2cnc(C)s2)=O)CC(NC(=O)Cc2coc3ccccc23)C(C2CC2)C1 CC1CC2CN(C(=O)C3CC3)CC2N1C(=O)CN1CCc2ccccc21 CCC(CC)(C(=O)N1CCC(O)(CN(C)C(c2nnn(C)c2N)=O)CC1)OC CCCCCC(O)CC(=O)N1CCOCC1C(C)(C)CNC(=O)CCS(C)=O C1(CC(=O)NC2(CC=CC(=O)NCC(CC)CO)CCC2)CCC=CCC1 C(N=c1cc(NCc2cn(C)nc2Br)nc[nH]1)c1cc(C(C)C)no1 N1(CC)CCC2=C(C1=O)C(c1ccc(Br)cc1Br)NC(=O)N2CCF c1(OC)ccc(NC(C2CCCCC2NC(c2cscc2Cl)=O)=O)nc1C C1(F)(C(=O)NCC(CNC(C(=Cc2cnc[nH]2)C)=O)(C)C)CCCCC1 Cc1cc(C(=O)NC(C2CCN(C(c3occc3C)=O)C2)C)cs1 c1(C(=O)NC2CCC(CNC(C3CC(OC)C3)=O)C2)cncc(F)c1Cl CCC(C)(O)C(=O)NC1CCN(C(=O)C=CC2CCCO2)CC1 C1(NC(c2c(C)[nH]cc2)=O)CCOCC1NC(C1CC1CC(C)C)=O C1(O)(CN(C)C(C2(C)CC2)=O)CCCN(C(C2(C)COC2)=O)C1 c1(C(=O)NC(c2cn(C)nn2)C(=O)N(CCC(F)(F)F)C)cc2cccn2cn1 N1(C(C(C2(O)CCC2)NC(CCCOC(C)C)=O)=O)CC(N(C)C)C(C)C1 N1(C(C2(SC)CN(C(COC)=O)C2)=O)CCC(F)(F)CC1 c1(COC)cc(CN2CCC(O)CC2C(=O)NCC2CNC(=O)CO2)cc(Br)c1 C(=O)(C1CCc2cc(F)ccc21)N(CCOCCN1CCN(C(C)=O)CC1)C C1(C)(C(=O)NCCCCCN(C(CCCCCC#C)=O)C)CCOC12CC2(F)F c1(SC)ccc(C(=O)NCCCCN(C(=O)C(O)C2CCCC2)C)cc1[N+](=O)[O-] C1(OC)CC2(C1)CC(C(N1CCCCC1CNCc1cncc(C)c1)=O)C2 C1(C)(C(N(CCCNC(C(C(=O)OC)C)=O)C)=O)CCCC1(F)F C1(CNC(c2cccc(C(F)(F)F)n2)=O)COCCN1C(=O)CSC(F)(F)F CC1=NOC(CCNC(c2cc(CCNC(=O)Cc3cnoc3)on2)=O)C1 c1(C(N2CCN(CC)CC2)=O)coc2c1CN(C(=O)CC1CC(O)C1(C)C)C2 c1(C(=O)NCC(CN(C(C=CCC)=O)C)C)nc(OC)ccc1C Cn1nc(C(N2CC(OCCNC(C3CCC3(F)F)=O)C2)=O)c2cc(F)ccc12 C#CCC(C)(C)C(=O)NC1CC(O)CN(C(=O)C(c2cnn(CC)c2)=O)C1 C1(CC(=O)NC2(CN(C)C(c3csc(-c4cnn(C)c4)n3)=O)CC2)CC2(CC2)C1 C1(C(=O)NC(CC=C)C(=O)N2CC(C#N)C2)CCC(C)(O)CC1 C1(NC(C(c2n(CC)ccn2)NC(C2(CO)CCCO2)=O)=O)CCC(=O)NC1C CC1C(NC(c2ccccc2-c2cccnc2)=O)CCS1(=O)=O C1(C(=O)Nc2nnn(CC(=O)OCC)c2C)C2Cc3cc(Cl)ccc3C12 N1(C(COCCCO)=O)CCC(N(c2ccccc2)S(C)(=O)=O)CC1 Cc1ccc(C(F)(F)C(=O)NC2CCC(CNC(C3C4CCCCC34)=O)C2)cc1 C(N=c1ccn2nccc2[nH]1)C1N(C(Cc2c(OC)ccc(C)c2)=O)CCC1 C1(NC(COCC=C)=O)CC2CCC1(NC(=O)C(N1CCSCC1)C)C2 C(N=c1nc(N2CCOC(c3nccs3)C2)c2c([nH]1)CCCC2)C1(C)CC(C)C1 C(=O)(C(CNC(c1cc(C)cc(F)c1)=O)CC(C)C)NCCCC(=O)NC C1(NC(C(CC=C)C)=O)CCCN(C(=O)CC23CCC(CC2)C3)C1C C1(C(N(C)Cc2c(C)cncc2)=O)CN(C(c2cn(C)cn2)=O)C(C)(C)C1 c1(CC)nc(C)[nH]c1C(=O)NCC1C2CN(C(=O)COC(F)(F)C(F)(F)F)CC12 C1(CNC(C2C(C(=O)OC)C2)=O)CN(C)CCN1C(C1(CCN(C)C)CC1)=O n1(CCOC)nnnc1C(C)(CCc1nccs1)NC(c1ccco1)C C1(CC)CN(C(=O)Cc2c(C)noc2C)CCC1NC(=O)CN1CCS(=O)CC1 C1(NC(=O)C=Cc2cccnc2)CCN(C(C2CC3(C2)CC(O)C3)=O)C12CCC2 N1(C(C(=O)NC)=O)CCN(Cc2snc(OC)c2Cl)CC1C(C)C C1(C(N2CCC(C(=O)N(CCC(C)(C)C)C)(OC)C2)=O)CC2(CC2)CN1C C(=O)(C(=O)N(CCC(=O)NCCc1nc[nH]n1)CCCO)N(C)C CC1CCN(C(C2CCSC2)=O)CC1C(=O)N(C1CCC1)C1CCC1 C(=O)(CC(O)CCC(C)CC)NC1(CC)CN(C(c2c(CC)occ2)=O)C1 Nc1cc(C(=O)NCCC2(O)CN(C(=O)COC3CC3(F)F)C2)cnc1Cl C1(NC(CC(C)(C)NC(C(C)n2ccnn2)=O)=O)CCC(=O)N(C)C1 N1(C(C(CC)SC)=O)CCCC(C(C)NC(C2(CO)CCOCC2)=O)CC1 Cc1ccc(C)n1CC(=O)N(CCCCNC(=O)CC1COC(CN)C1)C(C)C N1(C(C)=O)CCCC(O)(C(=O)Nc2ccc(C(=O)NC(C)Cn3ccnn3)o2)C1 N1(C(COC(CC)(C)C)=O)CCC(C(C)NC(=O)CO)C1 C1(CNC(C=C(COC)C)=O)CC2CCC1N2C(c1csc(C(C)(C)C)n1)=O C(=O)(C1=CCC(F)(F)CC1)NC1(CC)CCN(C(C2CC(SC)C2)=O)CC1 C1(NC(c2cc(Cl)cnc2O)=O)C2CC(O)C1N(C(c1csc(C3CC3)n1)=O)C2 N1(C(CCC(C)(C)F)=O)CCCC2CN(C(C3CC4(C3)CC3(CC3)C4)=O)CC12 C1(CC)OCCC1C(=O)NC(CC(=O)N(CCCCCO)C)C1CC1 C(N=c1[nH]nc(Cc2ccccc2)s1)C1(NC(CC=C)=O)CCOC1 C1(C(=O)NCCC2N(C(CCC(=O)N(CC)CC)=O)CCC2)CCCCS1(=O)=O C(c1ccc(Br)o1)=C(C)C(N1CC(C)(NC(=O)CN2CCCC2=O)C1)=O C1(C(=O)NC(c2ccoc2)C)CN(C(=O)C2=COCCC2)CCC1(F)F C12(C(N3CCCC(C)(NC(C(C)O)=O)C3)=O)CCC(C(F)F)(CC1)CC2 C1(NC(c2c(SC)ccn2C)c2n(CCCOC)nnn2)CC12CC(O)C2 N1(C(C2=C(C)CC2)=O)CC2CC1CC2NC(=O)C=CCN1CCCC1 c1(C(=O)NC(C2CCCCC2)CNC(CCC(=O)OC)=O)cn2cccnc2n1 N1(C(C(SC)SC)=O)CC2(C(=O)NCC(N3CC=CC3)=O)CCC1CC2 N(C(=NCc1sc(C)nc1C)NC1CCSC1)C1C(COC)C1 c1(C(=O)NC2CC(CNC3CCCO3)CC2O)cc(S(=O)(=O)N2CCCC2)c[nH]1 CC(C)CC(F)C=O.C1(c2cn(CC3(O)CCCC3(C)C)nn2)CNCC1(C)C C1(CNC(c2cc(C)sc2)=O)CN(C(c2cc(C(F)F)ccn2)=O)CCN1C c1(CCC(=O)NC2C(NC(CC3(CSC)CC3)=O)COC2)c(C)nc(S)nc1C CC(Cc1ccco1)C(=O)NC1(Cc2nn[nH]n2)COC1 c1(C(=O)OC)ncc(C(=O)NCC2COCC2NC(=O)C=C2CCCC2)s1 c1(OC(C)C(=O)NC2CC(Cn3cc(C4(C)CC4)nn3)C2)ccccc1Cl C=CCC(C)C(=O)N1CCC(NC(=O)CS(N)(=O)=O)C1C N1(C(C2CN(CCC)C(=O)C2)=O)CCC(CNC(=O)CCF)C12CCC2 C(=O)(C1CCC(=O)c2cccn21)NCC1C(C)CN(C(=O)CC2CCC(=O)N2)C1 n1(CC(=O)NCC(C)NC(C(CCSC)N(C)C)=O)ccc(O)nc1=O c1(NC(=O)OC)cccc2c1CCCC2NCC(C)COCCO Cc1cc(F)cc(NCC(=O)NCC(C(C)(C)C)NC(=O)CC2=CCOCC2)c1N N1(C(c2scc(C(C)=O)c2)=O)CCC(C)(C)C(CNC(=O)C(C)CN(C)C)C1 c1(C(CN(C=O)C2(C(=O)NCCO)CC2)O)ccc(F)c(Cl)c1 C=CCC(C)(CC)C(=O)NCc1ccc(C(=O)N(C2CCOCC2)C)cn1 C(=O)(CC(O)C(C)C)NCC1(CNC(c2ncc(OC)cn2)=O)CC(F)(F)C1 N1(C(CCOCCOCC)=O)CCOCC1CNC(c1cc(C)nn1C1CC1)=O C1(NC(C(=O)Nc2ccc(OCC)cc2)=O)Cc2nccnc2C1 Cc1ccc(CC(C)C(=O)NCC2CCCN2C(=O)CCc2scnc2C)cc1 C(CC(C(=O)N(C)Cc1ccc(C)cc1)NC(C1CC1(C)C)=O)SC c1(C(=O)NC23CC(CNC(C(CC)SC)=O)(C2)OC3C)cc2cccn2cn1 C(CCCCC(=O)N1CC(CS(C)=O)C1)N(C(=O)CCS(C)=O)C C1(CNC(c2c(C(=O)OCC)cccc2)=O)CCN(C(=O)C(C)(C)CF)CC1O N1(C(CN(C)C(=O)OC(C)(C)C)=O)CCN(C(=O)CCNC(=O)C=CCl)CC1C Cc1ccc(NC(=O)Nc2ccccn2)c(SC2COC2)c1 N1(C(C(C)(N(C(c2[nH]cc(C)c2)=O)C)C2CC2)=O)CCC2(C1)CC2(F)F CCCCS(=O)(=O)NC(C)C(N1CCC(NC(=O)COC(C)=O)C1C(C)(C)C)=O CCCC(CC(C)C)C(=O)N(CC(=O)NC(c1ccccc1C)C)CCC C1(N(c2ccccc2)C(C(=O)N(C2CCCC2C)C)=O)COCCN(CCO)C1 n1(NC(=O)C(F)(F)C2(O)CCC2)nccc1C(C)(C)C.C12CCC(C1)C(=O)N2C c1(C(C2(CO)CCC2)NC(CN(C(c2ccccn2)=O)CC)=O)ccccc1O Cc1ccc(C)c(OCC(=O)OCc2c(C(F)F)n[nH]c2C)c1 CCC(C)(CC)C(=O)NCC1CC(F)(F)CN1C(=O)CNS(=O)(=O)NC C(N=c1cc(C(N)=O)nc(C)[nH]1)C1N(C(C2CCC(CC)O2)=O)CCCC1C c1(-c2cn(CCN(C)C)nn2)ccc(C(=O)N(CC(=O)NCC#N)CC#N)cc1 C1(CNC(CCS(=O)(=O)NC)=O)CC2COCC2N1c1ncc(F)c(C)n1 N1(C(C(C(C)C)NC(c2cnn(C3CC3)c2)=O)=O)CC2(CNC(=O)C2)C1 Cc1cscc1C(=O)NCC(C1CC1)N(C(=O)Cc1ccc(Br)s1)C c1(C(N(C)CC2N(C(CCNS(CC)(=O)=O)=O)CCC2)=O)c[nH]c2cccnc12 CCC(C)CCC(O)CC(=O)N1CCN(C(=O)C(=O)OC)CC1 c1(C(=O)NCC2CCN(C(CCN(CC)CC)=O)CC2)n[nH]c2c1CCCCC2 c1(COC)nc(N(C)CC2CCCN(C(=O)CCn3cc(Cl)cn3)C2)cc(C)n1 C1(C(=O)NC(C)C(C)n2cccn2)CN(C(=O)Cn2cnnc2)CC1(C)C N1(C(Cc2c(C)nc[nH]2)=O)CCOCC1CCNC(C12CCC(C1)OC2)=O c1(NC(C2(CC=C)CCCN2C(=O)C(C)CCCOC)=O)cc(C)ccc1C c1(C(=O)NCCCN(C(c2c(C)cc(F)s2)=O)C2CC2)ccc2nccn2c1 C12(NC(c3cc(CCO)on3)=O)CCCC1CN(C(=O)Cc1ccno1)C2 Cc1cc(C(=O)N(C(C)C(=O)NCC2(CO)CCOC2)C)c(N)s1 C1(CC)CCCCC1OCCNC(CSC1CC(F)C1)=O c1(C(=O)OC)ccn(CC(=O)NC(C)CNC(C2CN(C)C2)=O)n1 CC1CCN(C(=O)CC(C)(C)C2CC2)CC1CNC(=O)CNC(=O)C(C)(C)C C1(CC(=O)NCC(CCOC)NC(=O)C=C(C)C(C)C)(CO)CCOCC1 CC(C)CC(C(=O)NC(C)CN(C(=O)CC1CCN(C)CC1)C)c1ccccc1 c1(OC)c[nH]c(C(N2CCC(NC(=O)C=Cc3ccc(C)cn3)C2)=O)cc1=O C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(=O)C(F)OC(F)(F)F)CCC1(F)F Nc1ccc(Br)c(C(=O)NC2CC(CNC(C3CCNC(=O)C3)=O)C2)c1 C1(C(=O)NCC(CNC(c2ccnn2CC2CCC2)=O)O)Cc2ccccc2O1 N1(C(Cn2ccc(C(=O)OC)n2)=O)CCC(F)C(NC(c2cc(Cl)c[nH]2)=O)C1 C1(NC(C23N(C(C(CCC)N(C)C)=O)CC(C)(C2)C3)=O)CC(C)(C)OC1(C)C N1(C(c2scc(C)c2)=O)CCC(O)C(NC(=O)Cc2sc(C)nc2C)C1 C1(CNC(Cc2c(C)occ2)=O)CCCC(NC(C2CC2c2cccnc2)=O)C1 C1(C(=O)NC2CC(NC(c3c(CCOC)n[nH]c3)=O)C(O)C2)CCC(=O)N(C)C1 C(=O)(NN1CCCC1C(N1CCCC(F)CC1)=O)c1ccc(COC)o1 n1(C(CC(=O)NCC(C)C)C)nc(C)cc1C.CCC1CN(C)C(=O)O1 c1(C(=O)NCC(CC(=O)NCCc2c(C)n[nH]c2)C)ncn2ccccc12 C1(C(=O)NC(CCC)C2CC2)(CNC(=O)CC2CC(OCC)C2)CC(C)(C)C1 c1(C(C)C)cc(C(=O)NC2CN(C(C3(C)CC4CC4C3)=O)C2)ccc1O CCC(C)CCCCC(=O)N1CC2CC1C2C(=O)N(C(C)CCC(C)C)C C1(O)(C(C)NC(=O)Cc2nncn2C)CCN(C(=O)CSc2nncs2)CC1 c1(C(C)(C)C#N)ccccc1CNCC(c1ccncc1)=O c1(Nc2nc(C)c(C(N3CC(F)(F)C3)=O)s2)cc2n(n1)CCCC2 C1(CC=C)(C(=O)NC(CNC(=O)C(=O)NC2CC2)CCC)CC=CCC1 c1(CNC(CC2C(CC)C2)=O)ccc(C(=O)NCC2(C)CCOC2)s1 C1(C(=O)NC2CCCN(C(c3c(C)cc(Br)o3)=O)C2)CC2OC(=O)OC2C1 c1(C(=O)NC(C)CCNC(C2(C)CCCC2(F)F)=O)n[nH]c2ccccc12 c1(C(=O)NCC(C)CNC(=O)CC(O)C2CCCC2)cc(C(N)=O)co1 C(=O)(C1CCN(C)c2ccccc21)NCC(C)NC(C1(COC)CCCO1)=O N1(C(C)=O)CCOCC1CCNC(N1C(C(=O)OC(C)(C)C)CC(C(=O)O)C1)=O NS(=O)(=O)c1ccc(F)c(C(N2CCC(C(=O)Nc3cnc(Br)cn3)CC2)=O)c1 CCC(CN(C)C)CC(=O)N1CCC(CNC(C2CCCCN2C(C)C)=O)C1 c1(C(=O)NCC2(O)CCN(C(C3C(C)(F)CCC3)=O)C2)ccnc2cc[nH]c12 c1(CC(=O)NC(C(=O)N(CCC(C)NC(N)=O)C)C)ccc(C(N)=O)nc1 c1(C(=O)NCCN(CCC)C(c2cccc(CC)c2)=O)ccc2nccn2c1 Cc1c(C(=O)NC(C)CN(C)C(c2cccc(-c3cc[nH]n3)c2)=O)ncn1C c1(C(=O)NC(C)CN(C(=O)COC2CC(F)(F)C2)C)ccc([N+](=O)[O-])cn1 C1(N(C)CC2(NC(C(CSC)O)=O)CCC2)CCN(C(=O)C(C(C)C)SC)CC1 C1(NC(c2cnns2)=O)C2CC(O)C1N(C(=O)Cc1cccc3ccccc13)C2 C1(NC(C2(CC)CC2)=O)CC2(C1)CC(C(=O)NCCc1c(O)n[nH]c1C)C2 C1(CN(C(=O)CC2CCSC2)C)CCCC1NC(C1(CCCF)CC1)=O C(=O)(C(O)CCC(C)C)N1CCC(N(C(c2c(CCC)n[nH]c2)=O)CCO)CC1 C(CCCC(C)SC)NC(=O)OC.C(=O)(C(C)CCN(C)C)NCCCOCCN C=CC(C)(C)CC(=O)N1C2CCC1C(CNC(C1(NC(C)C)CC1)=O)C2 N1(CC)CCOCC1C(=O)NC1CC1CCCC(=O)N1CC(c2nncs2)C1 C1(C(=O)NC2(CN)CN(C(=O)CC)C2)CCC(N(C)C)CC1.c1(C)ccnc(C)c1 c1(-c2cn(C3(NC(CN4C(C)(C)CC4)=O)CC3)nn2)cncc(C#N)c1 N1(C(COc2cncnc2)=O)CC2(CCC(=O)O2)C1.c12n[nH]cc1NC2=O c1(OC)cc(Cl)c(C(=O)NC2CN(C(C3CCCCC(F)(F)C3)=O)C2)cc1Cl C1(CC(N2CC3C(CN(C(C4(C=C)CCC4)=O)CC)C3C2)=O)CCCCC1(C)C CC1(C)C(C(N2CC=C(CNC(=O)CN3C(=O)CNC3=O)CC2)=O)CCS1(=O)=O C1(OC)CC2CC(NC(=O)C(c3cnn(C)c3)NC(=O)CC3CC(=O)C3)CC12 CCCC(C)(C)C(=O)NCC#CCNC(=O)C(C)(C)CCC C=CCCCCC(=O)N1CCOCC1C(C1CCC1)NC1CCC1 CC1(C)C(NC(c2ccc(Cl)cc2)=O)C2CCCN(C(=O)C(F)n3cccn3)C12 CN1CCN(C(C2(C3CC3)CCOC2)=O)CC(O)C1 C1(CNC(CN(C(COC)=O)C)=O)CCN(C(=O)COC(C)=O)CCC1(F)F C1(CN(C(C=CC(=O)NCC(C)CN(C)C)=O)C)COCCO1 N1(C(C(C)Nc2cccc(C)c2)=O)CCCC(C)(NC(=O)CSC2CC2)C1 c1(C(=O)NCC(C)N(C(=O)C2=CC(O)CCC2)C)c[nH]c2cc(F)c(F)cc12 C1(NC(C=Cc2ccc(C)cc2)=O)CCC(O)CN(S(=O)(=O)CC#N)C1 Cc1ccc(C(=O)NCC23CC(NC(c4cc(C)n(C)c4)=O)(C2)C3)c(Br)c1 C1(C(=O)NC2C(NC(C3(C)C(C)(C)C3)=O)CCC2)CCCCC1c1nc(S)n[nH]1 c1(C(=O)NC(C2CCCCN2C(C23CCC2C3)=O)C)ccc(OC2CCC2)nc1 c1(C(C)=O)nc(C(N2CCCC2CN(C(=O)CCC2CC(C)C2)C)=O)cs1 C(=O)(C1=CC2(CCOC2)C1)NCCOCCNC(C(C)S(N)(=O)=O)=O CC1CC(NC(=O)CCC=CBr)CCN1C(=O)CC1CC2(CC2)CO1 N1(C(CN2CCN(C)CC2=O)=O)CC2CN(C(=O)Cc3cc[nH]n3)CC2(C)C1 CC(=O)C(C)CC(C)C(=O)N1CCC1(C)CC(=O)NC12CCC(CC1)CC2 c1(C(N(C(CN(C(CC2N(CC)C(=O)CC2)=O)C)C)C)=O)cnc(C)c(C)c1 n1(CC(=O)NCC(CCNC(CC=C=C)=O)O)ccc(=O)n(C)c1=O C(=O)(C1=CCCOCC1)NC1C2(CCN(C(c3c[nH]c(=N)s3)=O)C2)C1 c1(C(CNC(C2(C(F)F)CCCO2)=O)NC(=O)OC(C)(C)C)ccc(F)cc1 C1(C)(NC(C(COC)NC(=O)CCc2ccoc2)=O)CCC(C)C1 C(N=c1[nH]c(=NCCC(C)F)c2[nH]ccc2[nH]1)c1[nH]nc(SC)n1 c1(C(C(N2C(CNC(CSCC)=O)CCCC2)=O)=O)c[nH]c2cc(F)ccc12 C1(NC(CC(=O)N(C)C)=O)CC2CC1CN(C(c1cnc(O)s1)=O)C2 c1(C(N(CCN(C(=O)CC2CCC3(CC3)CO2)CC)CC)=O)ccc(C)cc1C C1(C(=O)NC(C)(C)C2(CC3C(=C)C3)CC2)CCN(C(C2CCC(F)(F)C2)=O)CC1 C(=O)(CCCC(C)(C)C)N1CCCC(C)(CNC(c2c(C)oc(Cl)n2)=O)C1 C1(OC)CC2CCC(C1)C2C(N1C2CCC1CC(NC(=O)CC(C)SC)C2)=O C1(NC(C2CCCO2)=O)CC(NC(=O)Cc2ccco2)CC1O C(CC1CCc2ccccc21)N1CCC(NC(Cc2n(C)cnc2)=O)C(F)C1 C(c1ccccn1)=C(C(=O)NC(CC=C)CNC(=O)COC1CC(F)(F)C1)C Cc1c(NC2CCC(CN)C2)cnn1-c1ccccc1 N1(C(C2C(C(=O)NC(c3cc[nH]c3)C)C2)=O)CC(C)CCC1C C(=O)(CCC(=O)c1cccs1)NC(C1(O)CN(C(=O)C(=O)NCC2CC2)C1)C Cc1nc(Cc2cccc(O)c2)sc1C(N1CCC(N2CCOC2=O)C1)=O N1(C(CCCCN(CCCC)C)=O)CCN(C(=O)CC(C)C(F)F)CC1C1CC1 CC(F)(F)CCC(=O)NC1CN(C(c2cc(Br)c(C(F)F)s2)=O)CC1O N1(C(c2cn(CC(C(C)C)C)nn2)=O)CC(C)CC(C)C1.C12CN(CCO1)C2 C=CCC(CNC(=O)CCc1cc(C)on1)C(=O)N(CC)CC1CCCO1 C1(C2=CCN(C(=O)Nc3ccc(F)cc3C)CC2)(C(=O)OC)CCOCC1 Cc1ccc(F)c(CC(=O)N(CCCNC(=O)CCCOS(C)(=O)=O)C)c1 C(=O)(CCCCCCn1cc(CN2CC3CC3C2)nn1)N(CCCCO)CC Cc1cn2nc(C(N3CC(C(C)NC(c4nc(O)c(C)s4)=O)C3)=O)cc2c(=O)[nH]1 C1(C)(C(=O)NC(CNC(CN(C(=O)OCC)C)=O)C2CC2)C=CCCC1 c1(C(N2CC3C(NC(=O)CCCF)C(C3)C2)=O)cccc(S(F)(F)(F)(F)F)c1 CC1CCOCC1C(=O)NCCOCCN(C)C(c1ncsc1CC1CCC1)=O c1(C(N2CCC(O)(C(C)NC(CSCC)=O)C2)=O)ccc(Cl)cc1-n1cccn1 CC(C)S(=O)(=O)CC(=O)N1CCCC1CNC(=O)C(C)(C)Nc1ccccn1 Cc1cnc(C(N2CCCC(F)(CNC(=O)C(C)OCCC(C)C)C2)=O)c(C)c1 c1(C(=O)NCC2CCC(CC)C2)ccc(C(C)(C)C#N)cc1 Cc1cccc(C(F)(F)C(=O)NC2CC2CNC(C2COC(=O)N2)=O)c1 c1(OC)cc(C)nc(N2CCN(C3CN(Cc4cnc(Cl)c(C)c4)C3)CC2)n1 C1(C)(C(N(C(CCCC)C)C)=O)CCN(C(=O)Cc2cc(C)no2)C1 C(=O)(CC(C)CC(C)(C)C)N1CCN(C(CC(C=C)C)=O)C(C)CC1 C(=O)(C(CCCC#N)N1CCC(O)(CN(C)C)CC1)NCc1onc(COC)n1 C(=O)(C(C)(F)C(C)(C)F)NC1C2C(C)N(C(C(C)C)=O)C1C2 c1(OCCC)ccnc(NCCC2CCN(C(=O)CC3CCCCC3O)CC2)n1 N1(C(=O)CCc2ccc(Br)nc2)CCC2C1CCCN2C(=O)Cc1cncnc1 CC1CC(C(=O)NCC2CN(C(c3ccnc(CO)c3)=O)C2)C(C)O1 C1(C(N(CC(=O)NC(C#C)C(C)OC)C2CC2)=O)C2CN(C)CC12 C12CC13CCN(CC3)Cc1ccc(o1)C(=O)N2.C1(C(=O)NCCO)CC1(F)Cl N12CC3(CC(C3)C1=O)C2.N1(C(c2ccn(CC)n2)=O)CCCC(N2CCCC2)C1 C(=O)(C1=CCCCC1)N(CCCCC(=O)Nc1c(C(N)=O)nc(C)s1)C C1(CNC(C(CC)SC)=O)C(C)CCN1C(C1CC(C(F)(F)F)(OC)C1)=O N1(C(Cn2cccc(C)c2=O)=O)CC(C)CN(C(=O)C2=CCCC2)C(C)C1 C1(NC(CN(CCC#C)C)=O)CC12CCN(C(=O)C=CSCc1ccco1)CC2 C12(C(N(CCNC(=O)CCCC(F)F)CC)=O)CCCC(CCC1)C2O N1(C(C(c2cn(C)nc2)=O)=O)CCC2(NC(c3ccc(Cl)s3)=O)CC2C1 N1(CC(=O)NCC2CC(NC(c3ccnn3CC3CCC3)=O)C2)CCCC(O)C1 C1(NC(C2C(C)CC(C)O2)=O)CCN(C(c2cocn2)=O)CCC1CO C1(CC(=O)N(C(C)C(=O)NC2CN(C)NC2=O)CCC)CC(C2CC2)C1 c1(C(=O)NCCCN(C(CC2CC(OC)C2)=O)C)cn(CC)nc1C1CC1 C12(C(=O)NC3CC(NC(c4c(C)ccc(Cl)c4)=O)C3)CC1Cc1c[nH]nc12 c1(OC)cc(C(=O)NC2(CNC(C34CC3COC4(C)C)=O)CC2)ccc1F C(N=c1nc(N2CC(=O)NC(C)C2)c2c([nH]1)c(C)nn2C)Cc1n(CC)cnn1 c1(OCC=C)ccccc1C(=O)NC1CN(C(c2cccnn2)=O)CC1CCC=C N1(c2snc(CC)n2)CCCC(C2CC2NC(c2ccc3ncn(C)c3n2)=O)C1 C(C(O)CC(=O)NC(c1ccc(F)cc1)CNC(c1ncsc1C1CC1)=O)OC Cc1cc(C)nc(CC(=O)NC(C)CN(C)C(c2cc(C3CC3)ccc2F)=O)n1 C=CCCC(O)CNC(C1(NC(c2cnccc2C)=O)CC(F)(F)C1)=O C1(F)(CNC(c2c(OC)ccnc2)=O)CCN(C(=O)CS(=O)(=O)NC2CC2)CC1 C1(C2N(CC(=O)N(C)CCc3cc[nH]n3)CCC2)CCCN1Cc1ccccn1 CCCCC(O)CCC(=O)N1CCN(CCNC(C2COCCN2C=O)=O)CC1 CC(C)CCCCC(=O)N(C(CNC(c1c(Cl)cnn1C1CC1)=O)C1CC1)C CCCC(C(O)c1ccccc1)Nc1ccc(C(C)N)cc1 CCC(C)(C(=O)NC1CC2CCC1N(C(c1cncc(Cl)c1)=O)C2)C(N)=O CC(C)(CF)C(=O)NC(CNC(c1cnn(-c2ccc(Br)cc2)n1)=O)C1CC1 C(=O)(CC1=CCCCC1)N1CCC(CN(C(=O)CC2(N(C)C)CC2)CC)CC1 C1(NC(C=CCC)=O)CCOCC1NC(c1ccc(CC(=O)NCC)cc1)=O C#CCCC(O)C(=O)NCCCN(C1CCCC1)C(c1cc(CSC)no1)=O C1(COC)(N(C(=O)C(C)=C2CCC2)C2CC2)CCN(C(C2CCCCC2O)=O)C1 c1(C(=O)NCC=CCNC(C(C)OCC#C)=O)ncc(C(=O)OC)cc1Cl CCCC(C(=O)N1CCOC(C(C)C)C1)NC(=O)C=CCO N1(C(c2ccn(CC)c2C)=O)CC2CC(C(=O)NC3CCCCC3C)(C2)C1 C1(C)(C(=O)NCC(C2CC2)NC(C(C(C)O)(F)F)=O)COC(C)(C)OC1 c1(CN(C(C)CCO)C(=O)Cn2cncn2)ccc(I)cc1Br N1(C(c2ccc(C)[nH]2)=O)CCCCC1C1CCN(C(c2ncc(C)cn2)=O)C1 O=C1CCc2ccc(C(=O)NCC3CCN(Cc4ccc(Br)cn4)C3)nc2N1 c1(CC)nnsc1C(=O)NCC(F)CNC(=O)C(c1ccccc1)OC C1(C(C)C)C(=O)N1.C(CCC(=O)N1CCC1CNC(c1ccc(SC)o1)=O)OC C1(C(=O)NCC(C)CNC(c2noc3ccccc23)=O)CC2C=CCC(C1)C2 c1(C(=O)NC2(CCNC(CCCOC(C)C)=O)CCC2)cccc([N+](=O)[O-])c1N C1(CNC(C(CC)OC)=O)CCC(F)(CO)CC1.c1(C(=O)N)ccc[n+]([O-])c1 C(=O)(C(C)C(O)CC(C)C)NCCN(C(c1cc(C)cc(C(F)F)c1)=O)C N1(C(CN2C(C)CC2)=O)CCOC2CN(C(c3cc(CCO)on3)=O)CC12 Cc1cc(C)c(CN2CC(NC(=O)COCC3CCCO3)C(O)C2)[nH]1 c1(CNC(c2ncn(CC)c2)=O)cnn(C)c1C(=O)NCCC1CCC(C)C1 C1(CCNC(c2n(CC)nnc2)=O)CCCCN1C(=O)CCC1C(=O)ON=C1C C(CC1CCc2ccccc21)NC(=NCCOC)NCC1(C#N)CCCCC1 c1(OC)cncc(C(=O)NC(CO)C(=O)NCC(O)C(C)(C)O)c1 CCCCC(CC)NC(=O)CN(C(C)C(=O)NCC1CC1)CC#N.C(N)(=O)O O=C1CCCCN1CC1COCCN1Cc1cccc(Oc2ccccc2)n1 c1(CC)nnc2n1CCCC2C(=O)NC1CCC1NC(=O)C(C)CCCOC C1(CC(N2CCC(NC(c3ccoc3Cl)=O)C2C2CC2)=O)CC2CCC1CC2 Cc1nn(C)nc1C(=O)NCCC1CN(C(c2conc2C2CCC2)=O)CCO1 c1(C(=O)OCC)ccc(O)c(CNC23CC(C(=O)NC4CC4(Cl)Cl)(C2)C3)c1 C(C(=O)NC1(CNC(c2c(C)cccc2C)=O)CC1)(C(C)(C)C)OC N1(C(C(C)N2CCCC2)=O)C2CCCC1CC(NC(=O)Cn1cccn1)C2 c1(NC(C2CCC(CNC(Cc3cc(C)[nH]n3)=O)C2)=O)cc2cccn2c(O)n1 c1(C(=O)NC(C(=O)OC(C)(C)C)CS(C)(=O)=O)ccc(F)c2ccncc12 c1(C(N2CCC(C(F)F)(OC)C2)C(=O)NC2COC2)cn2ccc(C)cc2n1 c1(C(=O)NC2CN(Cc3c(C)scn3)CC2C#N)ccc2cccnc2c1 c1(CNC(C(c2cnn(C)c2)C)=O)nc(C(=O)NC(C)Cc2ccncc2)co1 C(=O)(C(C)P(C)(C)=O)N(CCNC(Cc1nc(OC)c(C)s1)=O)C(C)C C(C(=O)N1CC(CNC(C2CC(=O)N(C)C2)=O)C(C)C1)(C(C)C)OC N1(C(CC2CC(OC)C2)=O)CC(NC(C2(C)CC3CC3C2)=O)C(CC2CC2)C1 N1(C(c2c(C)con2)=O)CCC(C2CCN(C(c3cnc(F)cc3C)=O)C2)C1 C(=O)(C(CC)ONC(=O)C1CC1NC(=O)OC)NCC(=O)N(C)CC C1(CS(=O)(=O)OC)C(F)(F)C12CCOCC2.C1CCC1(C(=O)O)CO C1(C(=O)NC2(C)CCCN(C(C(C)C)=O)C2)CCn2nnnc2C1 c1(C(=O)NC(CCCC)CNC(=O)CNC(=O)C2CC2)ccc(C(F)F)cc1Cl CCC(CC)CC(F)C(=O)NC1COCCC1NC(c1c(C)ncnc1C)=O CCC(C(=O)OC)C(=O)N(C(C(=O)N(C1CCSC1)C)C1CC1)C c1(CC(N2CCCC2c2cn(CC3C4CCC3CC4)nn2)=O)ccccc1F c1(C(C)C)cc(C(N2CC(CC(C)NC(=O)C(C)O)C2)=O)c(C(C)C)[nH]1 c1(OC)ccc(OC)c(C(N2CCC(CNC(=O)C3=CCOC3)C(C)C2)=O)c1 c1(C(CC)CNC(C2(CNC(=O)COC(C)(C)C)CC2)=O)ccnn1C CCCCC(CC)CC(=O)N1CCOCC1CNC(c1cc2n(c1)CCOC2)=O c1(CSCCC)ccc(C(N2CC(N(C(=O)CCCC3CC3)C)C2)=O)o1 CN1C(=O)CC(C(=O)OCc2ccccc2OC(F)F)C1c1ccc(F)cc1 C1(C(C(C)C)NC(C(COC)OC)=O)CCN(C(=O)Cn2c(C)csc2=O)CC1 c1(C(N2CCOCC(CNC(c3n[nH]cc3F)=O)C2)=O)nccc2[nH]ccc12 C1(CC(=O)N(C2CN(C(c3cc(C#N)on3)=O)CC2O)C)CCOC(C)(C)C1 C1(CC(=O)N(C2C3CCCC23)CCl)CCCN(C(=O)Cn2cc(C3CC3)nn2)C1 C12CN(CC1(C)C)C2=O.c1(C(C)C)cccc(OC2CCCC2)c1 c1(NC)cncc(C(=O)NCC2(CCO)CCCC2)n1 c1(CC)ccc(Br)cc1C(=O)NC1CC(NC(=O)C(c2cnn(C)c2)=O)C1 C1(=O)C(C)N1.C(=O)(CCC1(C(=O)NCC)CC1)N.C(=O)NCC.SCC C(=O)(CCCC(=O)N1CC2CCCC2(NC(c2nccc3occc23)=O)C1)OC C1(C#CC(=O)N2CC(C)(NC(=O)CCc3nncs3)C2)(CC)CC1 C1(OC)(C)CCN(C(=O)OCC(=O)OC(C)(C)C)CC1.C(=O)(CCC(F)(F)F)N C1(NC(C(C)(C)CF)=O)CN(C(=O)Cc2cc(F)ccc2Br)CCC1CO CC(O)C(C)(C)C(=O)NC1CC(CCNC(c2ccnn2C2CCOCC2)=O)C1 c1(C(=O)NCCCCCCN(C(CC2C(C)C2)=O)C)nccc(N)c1Cl c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NC1CCN(C(=O)CC(O)C(C)C)C1 c1(C(=O)NCC2CC(NC(C(C)N(C)C)=O)CC2O)c[nH]c2cccc(Cl)c12 c1(C(N(CCNC(=O)CCc2ccoc2)CCOCCO)=O)c[nH]cc(Cl)c1=O N1(CCC)C(=O)CCC1C(=O)NCC(C)(C)CNC(=O)CSc1cccc(C)c1 N1(S(C(c2ccc(CN)cc2)C)(=O)=O)CCC(C(C)(C)C)(C(=O)OC)CC1 Cc1cnc2c(S(=O)(=O)NC3C4CN(Cc5ccccc5C)CC34)cccc2c1 C1(C(C)C)CN(C(=O)Nc2ncccc2O)CCN1S(=O)(=O)CC1CC1 C12(NC(=O)CC3C=CCC3)CCC(CC1n1cc(C3(O)CC3)nn1)C2 c1(C(N2CCCC(O)(C3CC3)CC2)=O)nnc2ccc(-c3ccc(F)cn3)cn12 N1(C(C2(NC(C3C(CC=C)CCC3)=O)CCCC2)=O)CCC(C=C)CC1 C(=O)(CC(O)c1ccccc1)N(C1CC(NC(=O)C(=O)NC2CC2)C1)C N1(C(C2CN(CC=CC)C(=O)C2)=O)CCC(C)C(CC(N(C)CP(C)(C)=O)=O)C1 C1(NC(C(c2ccc(OC)nc2)(F)F)=O)CN(C(=O)C(CSC)OC)CC1(C)C c1(OCC(=O)OC)cccc(NC(=O)CCNC(=O)COCC(C)(C)C)c1 C(C(C)(F)C(C)(C)F)NC(C1C2(CC(NC(C(CCC)C)=O)C2)C1)=O c1(C(N(C)CC2CCN(C(C=C(C)Cl)=O)CC2)=O)noc2c1CC(C)(C)CC2 c1(OCCOC)ccc(C(=O)NC(CNC(c2conc2C)=O)C2CCC2)cc1 Cc1cc(C(N2CCC(C(=O)NCCCC3CCCCC3)C2)=O)nnc1C c1(SC)cc(C(=O)Nc2cccc(NC(C3CCC(C4CC4)C3)=O)c2)cc(Cl)c1 C1(NC(CCCCC)=O)CCN(C(=O)CC2CCN(C(C)C)CC2)CC(O)C1 CC1(NC(=O)CCC2CCCCC2)CCN(C(=O)C=CC(=O)NC2CC2)CC1 Cc1cnncc1C(=O)NC1CCC(N(C)C(c2ccc(OC(C)C)cn2)=O)C1 c1(C(=O)NC2CC3CC(NC(COCC)=O)C3C2)c(C)nn2c(C)cc(Cl)nc12 N1(C(C2CC(CC)C2)=O)CC(O)CC1(C)C(=O)NCCCC(F)F C(=O)(C(CC=C)CC(C)C)N1CCC(Nc2cc(OC)nc(OC)n2)C1 Cn1c(O)nc2c(C(=O)NC3C4CN(C(C5(O)CCOC5)=O)CC34)cccc12 CC(O)C(F)(F)C(=O)NCc1nnc(O)nc1O Cc1ccc(C(=O)NCCC2(O)CCN(C(=O)C3=NOC(C)C3)C2)c(Br)c1 C1(N(C(=O)C(C)n2cncn2)CC)CCN(C(=O)CCCCNC(C)=O)CC1 C1(CNC(C=C(C)Cl)=O)(CO)CC12CCN(C(C1CC(CCO)C1)=O)CC2 c1(CC(=O)NCC2C(CNC(CCCSC(C)(C)C)=O)C2)ccc(S(N)(=O)=O)s1 c1(NCCN(C(CC2C(CC)C2)=O)CCO)ncc(C(N)=O)cc1Cl C#CCC(C(=O)N(C(C)(C(=O)NC(CC1CCCC1)CO)C1CC1)C)C1CC1 C12(CNC(c3ccc(CCC)cc3)=O)CCCN(C(c3ccncc3C)=O)C1C2 c1(C(N2CCC(C)(NC(C(c3ccccc3Cl)C)=O)C2)=O)c(F)ccc(N)c1F C1(CC(=O)N(C(C)CO)C2CC2)CN(C(C2CCOC2)=O)C(C)(C)C1 C1(C(=O)NCC2(NC(=O)CC3(n4ccnc4)CC3)CCC2)C2CC2C2CC12 C1(NC(COCC=C)=O)CC(C2CCN(C(=O)C(C)(C)CF)C2)C1 C1(C2CCN(C(c3ccc(C(=O)C4CC4)cc3)=O)C2)(NC(C(CC#C)C)=O)CC1 Cc1ccc(F)cc1-n1cc(C2CN(C(c3ccno3)=O)CCO2)nn1 NC(=O)CCCCC(=O)NCC1CCC(NC(=O)CCCc2ccc(O)cc2)C1 C(=O)(C1CCCc2sc(C)nc21)NCCN(c1nc(C(F)(F)F)ccc1Cl)CC C1(NC(CNC)=O)CC2(C1)CN(C(c1ccc(NC(=O)OC)cc1)=O)C2 Cc1cc(C(=O)NC2CCC(CNC(=O)CSc3ccc(Cl)cc3)C2)nc(O)n1 c1(C(N2CC=CC(NC(CC(CC)C)=O)C2)=O)cc2c(o1)CCCNC2=O c1(CC(=O)NC2C=CCN(C(CCCCC(C)C)=O)C2)cn(C)c2ccccc12 CC1CCCN(C(=O)Cn2cnnc2O)C1CCNC(c1cc(Br)no1)=O c1(C(=O)NC2(C)CN(C(C3CCC4(CCC4)CC3)=O)C2)ncc2ccccn12 N1(c2cc(OC)c([N+](=O)[O-])cc2)CC(C)CN(C(C)=O)CC1C N1(CC)CCOCC1C(=O)NC1(C)CCN(C(=O)CCCn2ccccc2=O)C1 C1(CN(C)Cc2c(C(C)C)noc2)CCN(c2nnc(C#N)s2)CC1 C1(CC)CC(C(N2CC(NC(c3cnn4ccsc34)=O)CC(C)C2)=O)CC(=O)N1 N1(C(C=C(C)Cl)=O)CCC2CN(C(=O)C=Cc3cccc(OC(F)(F)F)c3)CC12 c1(CC)nc(C(N2CCC(CCC(=O)NCc3nc(=O)o[nH]3)C2)=O)c(C)o1 Cc1[nH]nc(Cl)c1C(=O)NC(C)CCNC(=O)CCCn1ccnc1C c1(OC)ccc2c(C)c(C(=O)NC3CC(C)(NC(c4coc(C)c4)=O)C3)[nH]c2c1 CC1CN(C(=O)C2=CCCC2)CCC1NC(c1cc(-c2ccoc2)[nH]n1)=O c1(NC(C(c2cccc(OCC)c2)C)=O)cc(C)c(C(N)=O)c(C)n1 N1(c2cc(OC)nc(COC)n2)CC2(CC(NC(=O)C(C)C3CCCC3)CO2)C1 Cc1ncc(Cl)c(C(N2CCN(C(=O)CCc3ccc(N)cn3)CC2C)=O)n1 CCCC1C(=O)N1.c1(COC(C2(OC(C)C)CCC2)=O)ccc(N)cn1 c1(C(C)OC)cn(CC(C)NC(=O)C(CC)NC(C2CCCC2)=O)nn1 N1(C(c2cnc(CC)s2)=O)CCC(F)(C(=O)N(C)Cc2sccc2C)CC1 N1(C(C(C2CCC(C)(C)CC2)C)=O)CC2CC(C1)N(C(=O)C(=O)N=S(C)(C)=O)C2 CC1CCOCCN1C(C1CC(O)CCN1C(c1cccc[n+]1[O-])=O)=O c1(C(=O)OC)ccc(C(=O)NCC2(NC(C3CCCC3O)=O)CCOC2)c(Cl)c1 C1(NC(c2onc(C)c2C)=O)COC2(CCN(C(=O)CCN3CCCC3=O)C2)C1 CC1CN(C(C)C(=O)N2CC(CC(=O)NCCOCC(F)(F)F)C2)C1 N1(C(c2cocn2)=O)CCC(NC(C2(O)CCSCC2)=O)C(n2cccn2)C1 c1(C(N(C2CCN(C(=O)COCc3cc(C)no3)C2)CC)=O)cnnn1CC c1(C(=O)NCCN(C(=O)C(F)CC2CCC2)CCC)c[nH]c2cc(F)c(F)cc12 C1(NC(CCOC)=O)CCN(C(c2cc(C(C)C)c(O)cc2C)=O)C12CCC2 C1(NC(=O)COC2CC2)COCCC1NC(C12CC(CC(F)F)(C1)C2)=O C1(CC(=O)N(CCCCOC)C)CC2(C1)CN(C(=O)CCC1CC1)C2 C(CC1CCCC1)(C(=O)NCC1CCSC1)OC C(C(CNC(=O)CSc1cccc[n+]1[O-])C(F)(F)F)NC(C(C=C)(C)C)=O c1(NC(C2N(C(c3cn(CCC)nc3)=O)CCCC2)C)ncc2ccnc-2[nH]1 c1(-c2nc(NC(C=Cc3cn(CC)nc3)=O)on2)ccc(C#N)cc1 c1(C(C(=O)NCCC2CCCC2)NC(=O)OC)ccccn1 N1(C(CCN(C)CC)=O)CCN(C(=O)Cc2ccc(S(C)=O)cc2)C2(CCC2)C1 CCN=c1[nH]cc(C(N2CCCC2C2CC(NC(=O)C(C)CF)C2)=O)s1 N1(C(c2cc(C)n(C)c2)=O)CCCC2C1CCN2C(=O)Cn1nnnc1C1CC1 n1(CC)nc(C)c2cc(C(N3CC(CN(C)C(C4CC4C(F)F)=O)C3)=O)sc12 C12(CC)CN(C(=O)C(=O)NC3CCCN(S(C)(=O)=O)C3)CC1CCCO2 CCC(CC(=O)N1CCN(C)C(C(=O)NC(CC)CCO)C1)C(F)F c1(C(=O)NC2CCCC(NC(c3c(CC)cco3)=O)C2)cccc2[nH]ccc12 Cc1c(C(N2CCC3CCCC23)=O)cc([N+](=O)[O-])cc1Br O=C1CC(NC(C2(NC(C3CCCC3C(F)F)=O)CC2)=O)CC(=O)N1 C1(CC)C(C(=O)NCC(C)(C)NC(c2ncccc2C)=O)CCN1C c1(C(=O)NCC2C(NC(C(C(C)(C)C)OC)=O)CCC2)cc(S(C)(=O)=O)oc1C C1(C(=O)NCCN(C2CCCC2)C(c2cc(C)ns2)=O)Cc2ccc(F)cc2C1 Cc1nncc(C(N2CCCCCC2C(N2CCS(=O)CC2C)=O)=O)c1C c1(OC)ccc2c(n1)NC(C(N1CCC(O)CC(NC(=O)CSC)C1)=O)C2 c1(C(C)C)cccc(CC(=O)NC2CC2CNC(=O)CC2CCC(=O)N2)c1 c1(C(=O)Nc2c(NS(CCCC)(=O)=O)cccc2)cnc(Cl)c(C2CC2)c1 C1(O)(CCNC(c2nncc(C)c2)=O)CCN(C(C2CC(=O)N(C)C2)=O)CC1 C1(C(=O)NCCCNC(CN(C(CNC(C)=O)=O)C)=O)C2CCC3C(C2)CC13 c1(N(CC(C)CNC(C2(C(F)(F)F)CCCCC2)=O)C)nc(O)c2c[nH]nc2n1 c1(C(c2nnnn2C2COC2)NCC(N2CCCC2)C)ccc(Cl)nc1 Cc1cc(C(=O)N(C2CC(NC(c3cc(C)c(C)[nH]3)=O)C2)C)c(C)s1 N1(C(C=COc2ccc(C)cc2)=O)CC(C2CC2)C1NC(=O)OC(C)(C)C CON=CC(=O)NCCC1CCN(C(c2c[nH]nc2-c2ccc(Cl)s2)=O)C1 C#Cc1ccnc(C(=O)NCC2CC(C)N(C(C3CCC(N(C)C)CC3)=O)C2)c1 n1(-c2cn(CC)nc2)nc(-c2ccccc2CO)nc1C1CNC(=O)N1C N1(C(CC2(OC)CCC2)=O)CC(NC(=O)C(C)Cc2ccc(F)cc2)CCC1C Nc1ccc(CCC(=O)NC2(CC(=O)NCC3(CO)CC4CC4C3)CCC2)nc1 C(=O)(CCCCC(=O)OCCOC(C)(C)C)N(CCC#C)C Cc1ccc(-n2cc(C(=O)NCC(F)CNC(=O)COC3CCOCC3)nn2)cc1 CC1(C)CN(C(=O)C=CBr)CC(C)(C)C1NC(=O)CC1CCC1(C)C C1(NC(CCOCCOC)=O)CC(C)(CNC(=O)CC2(OC)CC2)C1 C1(C(N2CCN(CCCNC(C3CC4(CCC4)C3)=O)CC2)=O)(CC)CCNC1=O O(N=C1CCCCCC1)CC(N1CCOCC(CNC(CCS(C)(=O)=O)=O)C1)=O C1(C(=O)NCC=CCNC(C2CCCC(N(C)C)C2)=O)CC12CCCCC2 Cc1cccc(C(=O)NCCC2(O)CCN(C(=O)CCc3ccn(C)n3)C2)c1F C(=O)(CC(C)(O)COCC)NCC(C1CCC1)NC(C1(COCC)CC1)=O C1(CNC(c2cc(OC)nn2C)=O)CCCC2(CN(C(=O)CC3CC(C)C3)C2)O1 C1(C(N2CCCC(C(C)(C)OC)C2)=O)(NC(C(C(=O)OC)C)=O)CCC(C)(C)C1 CN1CC(NC(C2COCCN2C(c2cccs2)=O)=O)C(C)(C)C1 C1(C(=O)NCC(CN(C(=O)CC2COC(=O)C2)C)(C)C)Cc2c(F)cccc2O1 Cc1ccc(I)c(CNC(=O)NC23CC(C(=O)Nc4ccc(I)cc4)(C2)C3)c1 C1(C(N2CC(C)C(NC(c3ccn4ccccc34)=O)C2)=O)OC(C)(C)OC1(C)C C(=O)(C1CCCn2ccnc21)N1CC2CC(NC(C3CCOC3)=O)C2C1 CCCC(C(=O)NCC1(CNC(c2cnc(O)c(F)c2)=O)CC1)C(C)C C(=O)(C(F)(F)CCn1cc(CCCO)nn1)N(C(CCSC)C)C c1(C(=O)NCc2ccc(-c3c(O)cccc3O)nn2)ccc2c[nH]nc2c1 Cc1ccc(CNC(=O)N(CC(=O)NCC2(C)CCC2)C)o1 C=CCC1C(=O)NCC2(CCCC2)CCNC(=O)N1.C(=O)(CCS(C)=O)NC C1(C(N(CCCCC)CCO)=O)CC2(CCC2)CN1C(C1CCCSC1)=O C1(NC(C2CC(C)(C)CN2C(=O)CCc2nc(O)n[nH]2)=O)C2CCC(C2)C1(C)C CC1(CNC(C2CC3CCCC(C2)C3)=O)COCCN(C(c2ccoc2)=O)C1 c1(C(=O)C(C2(F)CCCOC2)=O)cccc(CN)c1.N1(C(=O)NCC)CC(OCC)C1 c1(C(=O)NCC2CC(NC(C3C(C=C)C3)=O)C2)ccc(CO)nc1 N1(C(=O)NCc2ccc(O)cc2I)CCC2(CCc3ccccc32)C1 C(=O)(CCCCCN(C(=O)CCC1CCCN1C)C)NC(C)C1CC1 CC(C)C(CC(=O)NCCN(C(=O)CCc1cncs1)C(C)C)c1ccon1 N1(C(C2N(CC)CCOC2)=O)CC2(COC(CNC(=O)CC(C)C(C)C)C2)C1 c1(OCCn2cc(CC(N3CC(N(C)C)C(O)C3)=O)nn2)ccc(O)c(CO)c1 N1(C(Cn2c(C)csc2=O)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C(C)C1C C(CCCC(=O)NCCC1(NC(=O)CCC(=O)c2ccc(N)cc2)CCC1)SC N1(C(C(C(C)C)SCC)=O)CCN(C)C(C(=O)Nc2ccc(O)c(F)c2)C1 C1(c2n(CC=C)nnn2)(NCC2(CCO)CC2)CCN(CC(=O)OC)C(C)C1 C1(CN(C(=O)CCCn2cccn2)C)CCN(C(=O)C(C)(O)c2ccccn2)C1 C(=O)(CCC(=O)NCCCCCN(C(=O)CNC(c1ccccc1C)=O)C)OC C1(NC(c2cc(CCC)on2)=O)CN(C(C2(CC)CCC2)=O)CCC1O N1(C(C)=O)Cc2cc(S(=O)(=O)NC3CNCC3c3ccccc3)ccc2OC1=O CC(C)(C(=O)N1CC2CCC1C(CNC(=O)CCCC(F)(F)F)C2)C(F)(F)F N1(C(c2c(C)[nH]cc2)=O)CCCC(CN(C(=O)CN(S(C)(=O)=O)C)C)C1 CC1(C(=O)NCC2(CNC(c3ccc(C(F)(F)F)s3)=O)CCC2)CC2CC2C1 C1(C(=O)NC(c2ccccc2)CNC(=O)C#CC(C)C)(OC)CCC(F)(F)CC1 N1(C(c2c(CCC)occ2)=O)CCC2(CC(NC(=O)COCC(C)C)CO2)C1 CC(C)(C)C(CNC(C1Cc2ccccc2C1)=O)C(=O)N1CCCCC(F)(F)C1 N1(C(c2ccc(NC)cn2)=O)CCCCCC1C(=O)Nc1cnncc1OC CC(C)(C)S(=O)(=O)CC(=O)NCC(C1CCOC1)NC(=O)CCC(F)(F)F c1(C(=O)NCC2C(CNC(C(c3c(C)cncc3)C)=O)C2)cc2c(ncn2C)s1 c1(C(N2CCC(C(C)NC(C3(C)CC(F)C3)=O)C2)=O)cccc(Br)c1Cl c1(C(N2CCC(F)(C(=O)Nc3cncc(C(N)=O)c3)C2)=O)ccnc(Cl)c1F N1(C(c2ccnn2C)C(=O)NC(C(=O)OC)C)CC(O)CC(O)C1 Cc1ccc2c(c1)SC(C(=O)NC1CC(NC(c3cc(C#N)no3)=O)C1)C2 N1(C(CC2(C#N)CC2)=O)C2CCCC1CC(NC(C1CCCCS1)=O)C2 CC1(CO)CCN(C(c2cc(Cl)n(Br)c2)C(=O)NCC2CC2)CC1 C(F)(F)(C(F)(F)F)OCC(=O)NCC1(F)CCC(NC(c2cnc(O)o2)=O)C1 C(=O)(C(C#N)C(=O)c1ccc(N2CC(C)OC(C)C2)cc1)NCCCOC c1(C(N2CCC(OC(F)F)CC2)C(=O)NCCCSCC)cnn2ccccc12 N1(C(C2COC(=O)O2)=O)CC2(CNC(C3(CO)CC3)=O)CCC1C2 C1(CNC(C2C(CC)CCN2C(=O)CCC(C)N(C)C)=O)OCC2CCC1C2 C(=O)(C1CCCc2nncn21)N1CC(NC(=O)CCOCC2CC2)CC2(C1)CC2 N1(C(CC2N(C(C(C)SC)=O)CCC2(C)C)=O)CCC2(CC(F)C2)C1 Cc1ccc(C(C)C)cc1C(N1CC(NC(=O)CC2COCCO2)C(C)(C)C1)=O CN1CC(C(=O)NC2CCCCN(C(C3(CF)CCC3)=O)C2)OCCC1=O C1(C(N2CCCN(CC)CC2)=O)C2CC(O)C(C2)N1C(C1CC2(CCC2O)C1)=O c1(C(N2C(CN(C(C(C(C)C)O)=O)C)CCC2)=O)c(F)ccc(C#N)c1F O=C(C1=C(F)CNCC1)N(C1CN(c2ccccn2)C1)CC1CCC1 C(=O)(NNc1ncnc2scnc12)Nc1cc(OCCC)c(C)cc1 C=CC1CN(C(=O)C(C)(O)C2CCC2)CC1NC(C1COCCOC1)=O Cc1cnccc1C(=O)NC(C1(CNC(C2CC23CCC3)=O)CC1)C c1(C(=O)NCC2CC(O)(CNC(=O)COC(F)(F)F)C2)snc2ccccc12 C12CCCCC1C(=O)NC2.N1(CC)CCCC(C(N)=O)C1.C1C(=O)NN1C C#CCC(CC(F)F)C(=O)NCc1cc(C)c(C(=O)NC2(CO)CCC2)o1 CC1=C(C(=O)N2CC(C(C)NC(C3CC(n4cnnc4)C3)=O)C2)S(=O)(=O)CCO1 C1(NC(C2(C)CC3CC3C2)=O)CN(C(C2CCCC2)=O)CCC1F C1(C)(OCCOC(CN(C(=O)CC2CCC3CC23)CC)=O)CCOCC1 C(=O)(C1=NOC(C)C1)N1CC(OC)C(C(=O)N(C)CCc2cccnc2)C1 c1(OCC(=O)NC2CC(N(C)C)C(O)C2)cc(Br)cc(F)c1F Cn1cc(C(=O)NC2CCN(C(C3OCCCC3(C)C)=O)CC2O)ncc1=O C(=O)(N=c1[nH]n(C)c2ccncc12)c1c(COC)ccs1 c1(OC)cnc(C(=O)NCCC(C)NC(C2CC2C2CCCO2)=O)cn1 O=C(O)CCC(=O)N(CC(c1ccccc1F)CO)Cc1nn[nH]n1 CCC(CC(=O)NCc1ccccc1CN(C(=O)CCOCC(F)F)C)C(F)F Cc1n[nH]c(C)c1C(=O)NCC1C(C)CCN1C(=O)C(=O)Cc1ccc(Cl)cc1 CCC(N=c1[nH]c2c(c(=NC(C)c3nnc(C)o3)[nH]1)CSC2)c1c(C)noc1C C(=O)(C1=CC2(CCOCC2)C1)NC(CC)CNC(C1(Cl)CC1(F)F)=O c1(C(=O)NC(C)C=CC(=O)NC2CC=CC2)ccn(C)n1 c1(N(C)Cc2cc(OCC)ns2)ccc(S(=O)(=O)NCCCCCCO)c(Br)c1 C1(C(=O)NCCCC(=O)N(C)C)C(C2CC2)CCN1C(c1cc(Cl)n(C)n1)=O c1(C2N(CC(=O)N(C(C)C)C)CCNC2)ccc(C2CC2)cc1F N1(CC)CCCC(OC(c2ccccc2)Cn2cc(CCC(C)(C)O)nn2)C1 c1(N(CC(C2CC2)OC)C)nc(=NCCC2(CCO)CC2)[nH]c2c(F)cccc12 c1(CC)cc(C(N2CCC(CN(C)C(C3(C#N)CCOC3)=O)C2)=O)cn(C)c1=O C12(C(N(C)CC3CCCS3)=O)CC(C(F)(F)F)(CO1)C2 C=C=CCCC(=O)NCC1CCN1C(c1cc(SC)c(C)o1)=O CC1CCN(C(C2CC=CC2)=O)CC1CNC(c1c(N)cccc1F)=O N1(C(c2ccc(C#N)cc2)=O)CC2C=CC1C(C(=O)Nc1cnc(O)c(F)c1)C2 c1(C(N2CCC(CCNC(=O)CCOCC(F)F)C2)=O)ccc(F)c(O)c1F C1(NC(c2cnsn2)=O)CC2CC(C1)N(C(=O)CN1CCOCC1)C2 C1(NC(c2scc(C)c2)=O)CS(=O)(=O)C2CN(C(=O)CN(C)C(=O)C3CC3)CC12 C(=O)(CCCCCC#N)Nc1c(C)ccc(C)c1.C12CC(C1)CNCC(=O)N2 CCC(C)(C)C(C)CC(=O)N1CC(NC(c2ncn(C(C)(C)C)n2)=O)CC(C)C1 c1(CC)cccnc1C(=O)N(CCCN(C(=O)C=C1CCC(C)CC1)C)C C1(c2c(F)cc(C(F)(F)F)cc2)CCN(N2CCC23CCCC3)C1 Cn1nnc(C(N2CCCCC2C(=O)O)=O)c1-c1ccc(-n2cccn2)cc1 C1(CNC(C(CC)F)=O)CCN(C(c2ccc[nH]2)=O)CCC1(F)F C1CS(=O)(=O)CCNC(c2cccs2)c2nnnn21.C1(CC)CCOCC1C c1(NC)ccc(C(N2CC(NC(C3(CF)CC3)=O)C3CC23)=O)cc1 c1(CN2C(CNC(N(CCCOC)CC)=O)CCC2)ccccc1 C1(C(=O)OCCSC(C)(C)C)CCCCN1C(C1CCCC1c1ccccc1)=O c1(C(N2CCC(N(C(=O)C(C)CF)CCC)C2)=O)c(C)cc(Cl)cc1C N1(C(c2c(C)nc(C)o2)=O)CC(NC(=O)CC2NC(=O)CNC2=O)CCC1C N1(C(C2(C(=O)OC)CC2)=O)CCC(C)(C(=O)NCCNC(=O)Cc2cccs2)C1 C(=O)(N=c1nc(SC)[nH]n1CCC#N)N1CC(CC)C12CCC2 C#Cc1ccc(CC(=O)NCC2(O)CCN(C(C3CS(=O)(=O)CCO3)=O)C2)cc1 C(C)(C)(CC(F)C(=O)NC1CCCCN(C)C1=O)NC(CC(=O)NCC)=O c1(C(N2CC(C(=O)N(C)C(C)C3CC3)(CC)C2)=O)c(C)cnn1C N1(C(c2cc(C)c(N)c(C)c2)=O)CC2(CCN(C(C3CC3Cl)=O)CC2)C1 c1(CNC2CCN(C(CCNC(C)=O)=O)C2)nc(C)c2ccccc2n1 C1(CCC)CN(C(C2CC3CCC(C2)O3)=O)CCN1C(=O)C(F)=C1CCCC1 C1(CNC(C=CSC)=O)CN(C(C2(C(=O)OC)CC2)=O)CC2(CCC2)O1 c1(CC)cc(=NCC2CCN(C(C3CC4CC4CC3C)=O)C2)[nH]c(COC)n1 C(=O)(CCCC(C)(C)NC(C1CCC(N(C)CC)C1)=O)Nc1c(CC)cccc1 c1(OCCNC(C23CCCCC2C3)=O)ccc(Br)cn1 c1(CC(N2C(C)CN(C(=O)CCC(C)CN(C)C)CC2)=O)cnn2c1CCCC2 c1(C(N2CCC(CCC(=O)NC(c3cnn[nH]3)C)C2)=O)ccn(C)c(=O)c1 c1(C(=O)NC(CNC(COC(CC)C)=O)C2CC2)ccn2ncc(Br)c2n1 C=CCN=C(NCCS(=O)(=O)CCC1CC1)NCC1CC(N(C)C)C1 Cn1ncc2ccc(C(=O)NCC3CC4CCC3N4C(c3cnns3)=O)cc12 C1(N(C)C(c2ccon2)=O)CCCC(NC(c2ocnc2C(F)F)=O)C1 Cc1c(CC(=O)NCC=CC(N2CC(CC(=O)N(C)C)C(C)C2)=O)ncn1C C1(C(=O)NCC2(CC)CC(C)(C)C2)CCCCCCN1C(=O)C(C)CC(N)=O C=CCCN=C(NCC1CCCC1OC)N1CCn2c(C(F)(F)F)nnc2C1 Cc1nn2cccnc2c1C(c1nnnn1C)NC1CCCCC1CN C12(CC(=O)NCc3ncccn3)CCC1CN(C(C1(SC)CCC1)=O)C2 C=C(Cl)CC(C(=O)NCC(O)COCC)NC(=O)CC(C)CC Cc1ccc(C(=O)N(CC(C)N(C)C(C2CCN(C)C2)=O)C)c(N)c1Br C1(C(=O)NCC(C)NC(=O)C=C2CCC2)NC(=O)CC1C N1(C(c2nccc(CC)c2)=O)CC2CCN(C(=O)C(C)(O)C3CCOCC3)CC12 c1(C(=O)NC(CC)(C)CNC(=O)COC)c(-c2cccc(OCC)c2)noc1C C=CC1(CO)CCN(C(C2CN(C(c3ccc(CC)nc3)=O)CC2(C)C)=O)CC1 CN1CCC2C(CCN2C(c2c(C(=O)N(C)C)nnn2C)=O)C1.C12(CC1)C(=O)NC2 c1(CN2C(C(=O)NCCOc3ccccc3)CC(O)C2)ccc(Cl)nc1Cl c1(CCC)nc(C(N2CC(CO)(NC(=O)C(C)C3CCOC3)C2)=O)co1 C1(C(N2CCN(C(C3CCCC3)=O)CC(CO)C2)=O)CC2(CCOCC2)CCO1 C(=O)(C(C)N=c1cc[nH]cc1)N1CC(NC(Cc2ccc(C)s2)=O)C(F)CC1 c1(C(=O)OC)cc2cc(S(=O)(=O)N(C)CC)ccc2o1.C12(CCOCC1)N(C)C2 N1(C(C2C(COC)C2)=O)CC=C(CC(=O)N2CC(C(=O)OC)C3(CC3)C2)CC1 C1(CC(C)C)CC(c2nnnn2C2CC2)(NC(CCO)C2CC2)C1 c1(CC)cccc(C)c1C(=O)NC1(C(=O)NCCOCCOC)CC(CO)C1 c1(C(=O)NC2C(C)N(C(C3CCC3)=O)CCC2)nnc2ccccn12 N1(C(c2cncc(NC)c2)=O)Cc2occ(C(=O)N(C)Cc3ccnn3C)c2C1 N1(C(C2CCCC23CC3)=O)CCN(C(=O)Cc2cc[nH]n2)C(c2ccccn2)C1 c1(OCC(N2C(C)(NC(c3ccnc(C4CC4)n3)=O)CC2)=O)c(F)cccc1F CCC(CC(=O)NCC1CC(CNC(c2cnc(O)c(Cl)c2)=O)C(O)C1)C(F)F N1(C(CCCCCOC)=O)CC2CN(C(=O)C(O)C(C)C)CC2(C)C1 CC(CN(C)C)CCC(=O)NC1CCN(C(c2cnsc2)=O)C1 Cc1cnc2n1C(C(=O)NCCN(C(=O)CN1CCC(C)C1)CC1CC1)CCC2 C(C)(C(=O)NCC(C1(O)CN(C(=O)Cc2nn(C)cc2Cl)C1)(C)C)(C(C)C)OC N1(C(CCc2ccc(C(C)=O)s2)=O)CCOCC1CNC(=O)COC1(C)CCC1 C1(NC(C(C)(C)c2cnsc2)=O)CC(F)CN(C(C2(F)CC2)=O)C1 Cc1ccc2cc(C(N3CCC(NC(=O)CC4(C)CCC4)C3)=O)[nH]c2c1 C1(N(C(c2cc(F)c[nH]2)=O)CC)CCCN(C(c2cnoc2C)=O)CC1 C1(CC(C)NC(CCCOC(C)C)=O)CCN(C(c2occc2C2CC2)=O)CC1 c1(C(=O)NC(c2ccc(CO)cc2)C(=O)OC)cnc(S(C)(=O)=O)s1 N1(CC(=O)NC(CNC(C(C2CC2)OCC)=O)(C)CC)CCC(O)CC1 C(CS(=O)(=O)CC(=O)N1CCOC(C(N)=O)C1)OC.c12c(cccc1C)C(=O)N2 c1(C(c2n(CCC)nnn2)NC2(COC)CCC2)cccc(CC#N)c1 C(=O)(C#CC(=O)N(C)C)N(CCNC(C1CCC(C)S1)=O)C1CC1 N1(C(C2CCCOCC2)C(=O)NCCCOC)CCCSCC1C c1(SC)ncc(CNc2cccc(OCC(F)F)c2)n1C C(C(C)(C(C)C)NC(c1cnc(O)s1)=O)NC(C1C(c2ccc(C)s2)C1)=O C(=O)(C1CCc2c[nH]nc21)NC(CN(C(c1c(C)nn(CC)c1C)=O)C)(C)C Cc1c(CC(=O)N(CCCNC(C(C)C(c2ccccc2)CC)=O)C)cnn1C C1(C(=O)NC(c2ccnn2C)CC)(OC)CCN(C(C2CCC3CC23)=O)C1 C1(C(C(=O)NCCC2(NC(C(=O)NCC)=O)CCC2)OC)CCCOC1 N1(C(Cc2ccc(C)nc2)=O)CCCC2(NC(C3CC3C3CC3)=O)CCCC12 C(=O)(C1=CC2C=CC1C2)NCC(CN(C(c1c(C)nn(C2CCOC2)c1)=O)C)C N1(C(C=C(C)CCc2ccccc2)=O)CC2CC1C2NC(=O)CCc1ccon1 CCC(C)(C)C(O)C(=O)NCCC(=O)Nc1ccc(C)o1 N1(C(=O)C=CC2CCOC2)CCC2CN(C(c3ccccc3O)=O)C2C1 C(C)(N=c1cc(C)nc(NC2CCOCC2)[nH]1)c1cc(C)c(F)cc1 c1(OCCOC)ccc(C(=O)NC(C)CCCNC(C2(C)CCOCC2)=O)cc1 CCC(C)CCCC(=O)N1CC(NC(C2CC(OC(F)(F)F)C2)=O)C(C)C1 c1(OC)cccc(C(C)C(=O)NCC2CC(O)CN2C(c2ccnn2C)=O)c1 N1(C(c2c(C(C)C)ocn2)=O)C2CCCC1CN(C(C1CC3(CCC3)CO1)=O)C2 C1(CN(C)C)CCCC(NC(C2(CNC(c3cnco3)=O)CCC2)=O)C1 C(CC(=O)N1CC(O)CC1CNC(c1csc2nccn12)=O)(C(F)(F)F)OC C1(C(N2CCC(C)N(C(c3n[nH]c(=N)s3)=O)CC2)=O)CC12CCC(F)(F)CC2 c1(N2CCC(c3ccc(CC)cc3)C2)nc2cccc(F)c2[nH]1 c1(OC)cc(N)c(C(=O)NC(CNC(C2CCCCC2(C)C)=O)C(C)C)c(F)c1 N1(C(c2ncn(CC)n2)=O)CCOCC(CNC(=O)CN2CC(C)(C)C2)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CCC2C1CCN2C(C1CCC(F)(F)C1)=O c1(C(N(CC(C)NC(CCCCC=C)=O)C)=O)ccc(F)c(C)c1C#N CC1CC(C)OC1C(N1CC(NC(c2cccc(N)c2)=O)C1)=O C1(CNC(CNC(=O)NC)=O)CN(C(c2cc(C3CC3)on2)=O)CC(C)(C)C1 C1(C(=O)NCC=CCNC(c2c(C(F)(F)F)ncn2O)=O)CCC2CC1CO2 c1(C(=O)NCCN(C)C(C2(F)CC=CCC2)=O)ccc2c(c1)CCCO2 Cc1cnc(C=CC(=O)NC2COCC2NC(c2ncoc2C(F)(F)F)=O)[nH]1 C1(CNC(C(C(C)C)NC=O)=O)CCCCN(C(=O)C=C2CC2)CC1 CN1CCN(C(C2CN(C(C3(C)CCCOC3)=O)C2)=O)CC1CNC(N)=O c1(C(=O)NCC(CO)C2CC2)coc2c1CN(C(=O)C(O)CC(F)(F)F)C2 n1(CCC(C)C)ncc2cc(C(=O)NC3COCCC3NC(=O)CCF)cnc12 C1(C(N(C2CCC(C(N)=O)CC2)C)=O)CN(C(=O)CC2CCCNC2=O)CCO1 Cc1nc(C(F)(F)F)ccc1C(=O)NC(C)C(C)NC(c1csc2nnsc12)=O Cc1ccc(CC(C)N(C)C(c2csc(-c3cnn(C)c3)n2)=O)cc1 C1(C(=O)NC2(C(=O)NCC)CC2)(CF)CCN(C(C2CC3CC3C2)=O)C1 O(N(C)C(=O)C(NC(=O)CC1CSCCO1)SC)CCCC(=O)OC S(=O)(=O)(c1ccc(I)cc1F)NC(C(C)(F)c1ccccc1)=O N1(C(c2sc(C)c(O)n2)=O)CCCC(CNC(C2CCC3(CC2)CC3)=O)CC1 N1(C(CCSCCC)=O)CCC(C(=O)NC2CC(C(F)(F)F)(OC)C2)C(CC)C1 c1(C(N2CCCC3CCN(C)CC23)C(=O)NCCOC)nc2ccccc2nc1C N1(C(c2c(C)oc(C)c2C)=O)CCCC(C)(C)C1C(=O)NCC1CC12CC2 C(c1cn(C2CN(C(C3CC(C)(C)CO3)=O)C2)nn1)=CC Cc1cn2c(n1)CCC(C(=O)NC1CCCN(C(c3cnc(C(C)C)s3)=O)C1)C2 C1(NC(CCc2ccc(OC)cc2)=O)CC2CC1N(C(c1cc(CO)[nH]n1)=O)C2 n1(CC(CC)CC)nc(-c2cncnc2)nc1-c1ccsc1Cl c1(CCNC(N2CCC(c3cccnc3F)C2)=O)ccn2ccnc2c1 N1(CC(=O)NCCN(CC(C)O)C(=O)CC2CC2C(F)(F)F)CCOCC1=O C(=O)(CCCC(C)(C)C)N1C(C)(C(NOCCC(C)O)=O)CCC1 C(C)(C)(CCCNC(=O)CC1C=CC(NC(=O)CNC2CC2C)C1)OC N1(C(=O)NCc2n(CCC)ncn2)CCN(Cc2ccccc2)C(=O)C1C c1(NC(C2(O)CCN(C(CCC=C(C)C)=O)C2)=O)cc(Br)cc2[nH]ncc12 C#Cc1ccc(CC(=O)N(C2CC3CC2N(C(=O)C=C(CC)CC)C3)C)cc1 CC(CO)CCCNC(=O)CSCCNC(C1OCCC1(C)C)=O c1(C(=O)NC(CNC(c2cc(SC)oc2)=O)C2CC2)ccc(Cl)c(N)c1 N1(C(Cn2c(C)ncc2)=O)CCC=C(C(=O)N2CCC(C3(C)N=N3)C2)C1 c1(NC(=O)OCC)ccccc1C(N1CC(C)(NC(=O)CSC(F)(F)F)C1)=O N1(C(C(CC)N2CCCC2)=O)CCCCC(C(=O)Nc2cccc(F)c2C)C1 c1(C(=O)NCC2C(NC(CN(S(C)(=O)=O)C)=O)C2)ccn2c(=N)[nH]nc2c1 N1(C(c2c(CC)nc(C)nc2)=O)CCC2CN(C(c3cn(C)nc3SC)=O)CC12 C1(C(=O)NCCCN(C(=O)CC2CC2(C)C)C(C)C)CC12CC(C)(C)C2 N1(C(C=CC(CC)C)=O)CCOCCC1C(=O)NCc1cccc(OC)n1 C1(C(C(=O)NCC(C)(C)OCCNC(C(F)OC)=O)O)CCCCCCC1 C1(NC(C(CC)n2cncn2)=O)CCC(N=c2[nH]c(C#N)c(Cl)s2)CC1 N1(C(C(=O)NCCCCNC(C(C)Cc2cnn(C)c2)=O)C)C(=O)CCC1=O N1(C(C(C(CC)C)O)=O)CCCC2(NC(=O)Cc3ccc4c(c3)CCO4)CC2C1 C#Cc1ccc(C(N2CCC(O)(CC3CC3)CC2)C(=O)NCC(F)F)c(F)c1 C1(C(N2C(CNC(C3(C)CCCS3(=O)=O)=O)CCC2)=O)CCCC12OCCO2 n1(CC(=O)N(CCCN(c2nncs2)C)C)cnc2ccccc12 C(CCC)(CCCNC(=O)CN1CCCNC1=O)NC(C(CC)NC(C)=O)=O C1(NC(CSCC)=O)CN(C(c2cc3c(cc2O)OCO3)=O)CC2(CCC2)C1 N1(C2CC2NC(c2cccnc2)=O)CCC(C(=O)NCCNC(=O)OCC)CC1 n1(CC(=O)OC)cnc2ccccc12.C1(=O)CC(C(=O)O)N1C1CC1 C1(CNC(CCCC)=O)CN(C(C2(C)CC(O)CN2C)=O)CC1(F)F N1(C(N2CCC(O)(C3CC3)CC2)=O)CCC2(CC1)Cc1ccccc1C2=O C#CCCC(O)CCNC(c1cnc(CNC(=O)C(C)n2ccnc2)nc1)=O C1(OC)CC(CC(=O)NCCN(C(=O)C=CC2CCC2)C(C)C)C1(C)C N1(Cc2n(C)cc(Br)n2)CCC(CNC(c2cc(Br)cnc2Cl)=O)C(F)(F)C1 N1(Cc2cnc(CCC)s2)CCN(C(C2CN(C)CCO2)=O)C(CC)C1 N1(C(C=Cc2nc(C)sc2)=O)CCCC(NC(C2CCS2(=O)=O)=O)C1C C1(CCC)CN(C(c2ccc(C)c(C)c2)=O)CCN1C(=O)CN1CC(C)(C)C1 c1(NC(=O)CCc2cccnc2)ccc(C(N2CCC2)=O)cn1 C(=O)(C1OCCn2ccnc21)N1CCCC(CC=C)(NC(=O)Cn2nccn2)C1 CCCN=C(NCCC(=O)OCC(C)(C)C)N1CCC(F)(c2ccc(F)cc2)C1 CCC(CCC(=O)NCC(C)S(C)(=O)=O)NC(c1cn(CC)cn1)=O C12CCCN1C2=O.c1(C(=O)N)ccccn1.CC1(C(=O)NC2(C)CC2)CCC1 CC1CN(C(C2CCC(N(C)C)C2)=O)CCC1CNC(=O)CCc1ccccc1 C1(CC(N2C3CC(CNC(c4cnns4)=O)C2CC3)=O)CNc2ccccc2O1 c1(C(=O)NC(C(C)(C)NC(c2c(CC)cco2)=O)C)cccc2c1CCC2 c12cc([nH]n1)N2.N1(C(CCN(CC)CC)=O)CCC(OCC(C)C)C1 c1(C(N2CC(CS(C)(=O)=O)C2)=O)c[nH]nc1SCCC(=O)NCC1CCCC1 C1(C(N(C23CC(CC(C)C)(C2)C3)C(=O)CN(C2CCCC2)C)=O)CCCN(C)C1 Cc1ncc(N)cc1C(=O)NC(C)(CNC(=O)Cn1ncn(C)c1=O)CO N1(CCN(C(=O)CCN(C)C(c2ccsn2)=O)C)CCOCC1 Cc1ncnc(C(=O)NCc2nn[nH]n2)c1C Cc1ccc(CCNC(C2CC=CCC2)=O)c(F)c1 C1(C(N(CC(O)CF)C)=O)CC2(CCC2)CN1C(c1cc([N+](=O)[O-])c[nH]1)=O c1(C(C)=O)nc(C(=O)N(C)CC2CCN(C(=O)CC3CS(=O)(=O)C3)C2)cs1 C(C(CN=c1nc(C(=O)NCC2(COC)CC2)cc(C)[nH]1)C(F)(F)F)OC N1(C(C(C)NC=CC(F)F)C)CCN(C(C)(C)C)CC1.N(C)C C(C)(C)(CCC(=O)NC1CC2CCC(C1)O2)NC(C(CCC)=CCC)=O c1(C(N2CC(C)(CC(=O)NC(C)C(=O)NC3CC3)C2)=O)c(F)cccc1Cl CCCCCCCC(=O)NCC1CCCCC1NC(=O)Cn1ccnn1 C1(C(=O)NCCCNC(c2c(F)ccc(F)c2Cl)=O)CCc2nc(O)[nH]c2C1 C1(C2CCN(C(C3CC(C4CC4)=NO3)=O)CC2)(NC(c2c(C)ncnc2)=O)CC1 c1(C(=O)NCCCC(C)(C)NC(=O)C(O)Cc2ccccn2)ccc(N)c(F)c1 C(C(C)(C)C(=O)NCC1CN(C(=O)CCc2nc(C3CC3)no2)C1)OC CC1(C)CN(C(C2COC3(C2)CN(C(C2CC2C(C)(F)F)=O)C3)=O)CCCO1 N1(C(c2cccc(OCCC)c2)=O)CCC2(NC(c3cc(C)no3)=O)CC2C1 C(=O)(C1=C(C)CCOC1)NC(CCCC)CNC(=O)Cc1cnccc1Cl N1(C(C(C2CCC2)OCC)=O)CCC2(CCCN2C(=O)C=CC2CCCO2)CC1 c1(C(=O)NCC2(CNC(C3(CC#C)CCCCC3)=O)CC2)cc([N+](=O)[O-])c[nH]1 C1(CNC(C2(OC)CCOC2)=O)COCCN(C(=O)C(C)N2CCC2)C1 C=CCCCCCCC(=O)N1CCC2C(CCN2C(=O)CC(O)C(C)C)C1 C1(NC(C(C)SC)=O)CCOC12CCN(C(C1CC(OC)(OC)C1)=O)CC2 c1(NCCC(C2CC2)OC)nccc(N2CCC(NCC(=O)OC)CC2)n1 N12CC(C(C3CC3)C1)C2=O.C1(COC)CC(C(=O)NC2(C(O)CO)CC2)C1 N1(C(c2c(OC)csc2)=O)CCCC(CNC(=O)COCc2cc(C)on2)CC1 C1(NC(C2N(C(C)=O)CCCC2)=O)CCC2CCN(C(=O)COCC(F)F)C1C2 C1(NC(CC2C(C)CC2)=O)CC2(CCN(C(=O)C(C)(C)N(C)C)C2)C1 C(C1CCCc2nccn21)NC(=O)NCCOC(c1c(OC)ccs1)=O Cc1nonc1CC(=O)NC1CCC1C(=O)N(C1CC2(CC2)C1)C c1(C(=O)OC)ccc(C(c2nnnn2CC2CCCO2)NC(C)(C)CF)s1 C1(NC(c2c(CC(C)C)sc(Cl)n2)=O)CC2CC(NC(=O)COCCF)CC2C1 Cc1nc(N2CCN(C)CC2CNC(=O)C(c2ccnn2C)O)c2ccsc2n1 N1(C(Cn2c(C)ncc2)=O)CCCCC1CCNC(=O)C(C)(C)n1ccnn1 C1(NC(C2C(C)(C)C2(C)C)=O)CN(C(=O)C2=NNC(=O)CC2)C2(CCCOC2)C1 CC(C)CC(C)C(=O)N1CCC(N(CCO)C(C2COC(C(F)(F)F)C2)=O)CC1 c1(C(=O)NC2CN(C(C3(F)CC3)=O)CCC2F)cc2cccnc2o1 c1(CNC(=O)NCC2CN3CCCN2CC3)cn2cc(Br)ccc2n1 Cc1nc(C(=O)NCCCOCCOCCNC(C2(C)COC2)=O)[nH]c1C N1(C(CS(=O)(=O)NC)=O)CCN(C(=O)C(C2CCCCC2)O)C2CCCCC2C1 C12(CNC(C=C(C)C(F)F)=O)CC1CN(C(c1csc(Cl)n1)=O)C2 CC#CCC(CO)NC(=O)CCN(C(C1CCCCCC1)=O)CC CCC(CC)(CCNC(C1CCCC(O)C1)=O)NC(c1cc(C(F)F)no1)=O C(=O)(CCCCC(C)(C)C)N1C(CC(=O)NCCCS(C)=O)CC2(CC2)C1 N1(C(C(C)OC)=O)CCCC2(CCN2C(=O)C(n2nc(C)cc2C)C)C1 CCC(CC)C(C)C(=O)NC1CCC1NC(c1ncoc1-c1cnn(C)c1)=O C1(C(=O)NC(CNC(c2ncc(C)cc2O)=O)CC(C)C)CCC2CCCCN12 C(CC(=O)NC1CC2C(NC(C3(C)C=CCC3)=O)C2C1)(C(C)C)OCC c1(NC(=O)NCC2(C)CCC(CC)CC2)ccc(OC)cc1N=[N+]=[N-] C1(NC(=O)CCc2ccsc2)CCC(O)CN(C(=O)CN2CCCS2(=O)=O)C1 C1(C)(C(N2CC(C(C)NC(=O)CC3CCSCC3)OCC2)=O)CCS(=O)(=O)CC1 C1(CC(N2CC3C(CNC(c4cnc(C)n4C)=O)C3C2)=O)CCCCC12CC2 CC(C)(C#CC(=O)N1CC(N2CCCC2)C1)CNC(c1cnc2ccccn12)=O c1(N(C2CCN(CCO)C2)C)ccn2ncc(S(=O)(=O)NCCC3CCC3)c2n1 C=CCCCCCC(=O)N1CC(CN(C(=O)C(C)C(O)CC)C)C1 N12CC(C3CC13)OCC2=O.N1(C(CN(C(=O)OCC)C)=O)CC(F)(CSC)C1 C1(C(=O)NC(c2ccncc2)(C)C)CCCN(C(C2CCCN2C2CC2)=O)C1 C(c1c(Cl)cccc1Cl)=CC(=O)NC1CN(C(C2CC(C#N)C2)=O)CC1O C(=O)(C1=COCCC1)N1C(C(=O)NCc2cc(COC)on2)CCC1C1CC1 N1(C(C(C2CCC2)OC)=O)CCOC(C(=O)NCCC2CC(C)=NO2)C1 C(C1CN(C(=O)CC2(O)CCCC2)CC1C(=O)NOC(CO)C(C)C)=CC C1(NC(C2CC(C)SCC2)=O)CCN(C(c2cc(O)nn2C)=O)CC1F N1(C(Cc2c(Br)cn(C)n2)=O)CCCCC(NC(C2(C)CC=CCC2)=O)C1 C#CC1(F)CCN(C(C2C3CC3CN2C(=O)C(C)OC)=O)CC1 C(=O)(N=c1[nH][nH]c2cc(F)ccc12)NC(Nc1ncnc(N(C)C)c1Cl)=S C=C(C)CCCC(=O)Nc1ccc(NC(c2ccsc2C#N)=O)cc1C C(=O)(C1=NOC2COCC12)NCC1(CNC(CC(CCC)C)=O)CCCC1 CC(C)CC(F)C(=O)NC1CCCCC1NC(=O)CSc1ccccn1 N1(C(CC(C)C2CC2)=O)CC2(CO)CC1(C(=O)NCC1CC13CCCCC3)C2 c1(C(N2CCC(O)(CCNC(C=CC(CC)C)=O)C2)=O)cc(C)cc(C)c1N Cc1ccc(NNC(=O)CSCC2(O)CCOCC2)c(C)c1 c1(OC)cnc(F)c(C(N2CC(CCNC(C3C4CC4C4CC34)=O)(OC)C2)=O)c1 c1(CC)ccc([N+](=O)[O-])cc1C(N1CCOC(CCNC(c2cc[nH]c2)=O)C1)=O N1(C(CCN(C)C(C2CCOC(=O)CC2)=O)=O)CCCC(O)(CO)C1 C1(NC(C)=O)CCCCCN1C(=O)CS(C)(=O)=O.c12cccc(c1)CO2 CC(CS(C)(=O)=O)C(=O)N1CC2CCC1CC2NC(C1(CO)CC1)=O c1(C(=O)NCC(C)NC(c2ccns2)=O)csc(-c2ccoc2)n1 Cn1nc(CC(N2CCCCC2CCNC(=O)C=C2CC2)=O)c2ccccc12 N1(C(C2N(C(c3cc(OC)c(C)cc3)=O)CC=C2)=O)CCCC2(CCOC2)C1 c1(C(=O)NC2(CNC(c3cc(N)cc(F)c3)=O)CCC2)c[nH]c2nccc(Cl)c12 C(=O)(C1CCCc2nc[nH]c21)NCCCOCCNC(C(CC)SC)=O C(=O)(CCCC(C)(F)F)NC(CC(C)NC(c1n(CC)ccc1)=O)C N1(C(c2cc(OC)c(F)c(OC)c2)=O)CC2CC(C1)CN(C(=O)CCCCBr)C2 c1(C(N(CCCNC(CC(C=C)C)=O)CC)=O)ccc(O)c(CO)c1 N1(C(C23N(C(C(C(C)C)OC)=O)CCC2C3)=O)CCC2(CCC2)CC1 C1(C(=O)NC(CC)(CO)CO)CCCN(C(c2ccc(C(C)C)cc2)=O)CC1 S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(C(=O)NCCCCC#C)CC1 N1(N(CC(F)F)C)CC2(CCCN(C(=O)C=O)C2)C1.C12(C=O)CCC(C1)C(C)(C)O2 C1(CNC(CN(C)C)=O)CC2CCC1N2C(c1ncc(C(F)(F)F)s1)=O C1(C(=O)NC(c2ccccc2)CCC)NCCC1C1CCC1 Cc1ccc(C(=O)NC2CCN(C(C3CC(=C4CC4)C3)=O)CC2CO)cc1F CN1C(=O)NCC1C(=O)NC(c1ccccc1)CNC(C12CCCC1C2)=O CC1CCN(C(=O)CC2CN(C(C3CN(C(N)=O)C3)=O)CCO2)CC1(F)F C1(CN(CC(=O)NCCCOCC)CCOCCO)CCCC(=O)C1 C(C)(CCC(=O)NC(CNC(=O)CNC(C1CCC1)=O)C(C)(C)C)SC c1(C(=O)OC)ccc(C(=O)NC2(CNCc3ncc[nH]3)CCC2)n1C n1(CCC)cc(C(=O)NC2CCC(CNC(C3CCCC(COC)O3)=O)C2)nn1 C1(NC(C(COC)CC)=O)CN(C(=O)C=NOC)CCC1(C)C c1(C(=O)NC2CC(C(C(=O)NCCCC(=C)C)F)C2)ccc(F)c(C)c1 C12(NC(c3ccc(OC)cn3)=O)COC(C1)C(NC(=O)C=Cc1ccc(C)o1)C2 N1(C(C(COCC)C)=O)CC(C(N2CCC(COC)C2)=O)CC(C)C1 c1(CNC(C=CC(CC)C)=O)cc(C(N2CC(OCCO)C2)=O)ccn1 c1(CC)ccc(C)c(C(N2CC3CC(N(C(=O)C(C)(C)CC4CC4)C)C2C3)=O)c1 C(=O)(C(C)(C)C(F)c1ccccc1)N1CC(NC(C2C(C)(CC)C2)=O)C(SC)C1 C1(C(C(=O)NCCCOC=C)NC(c2cscn2)=O)CC=CCC1 N1(C(C2C(C)OC(C)C2C)=O)C2CCC1CC(CNC(C1(C)CCCO1)=O)C2 C=C1CCN(C(=O)CC(C)n2cccn2)C(C(=O)NC2CCCC2CF)C1 c1(C(N2CCCCC2c2ccc(Cl)nc2)C(=O)NC2CC2)cc(Cl)c(Br)cc1F N1(C(c2cc(C)no2)=O)CCC(NC(=O)C(C)(C)CCF)C(C)C1 c1(NC(CC2C(CNC(c3ccc(OC)cc3)=O)C2)=O)cnc(OC)cc1C C(=O)(C(CC)C(C)C)NC(CNC(c1cncc(C(=O)OC)c1)=O)CCOC N1(C(C(C(C)C)SC)=O)CC(CNC(c2ccc(C(N)=O)s2)=O)OC(C)(C)C1 N1(C(CNC(CNC(CCC(CC)OC)=O)=O)=O)CC2NC(=O)OC2C1 c1(C(C(=O)NCCCC2CC2)N(C)CCc2cccc(O)c2)nccc(Cl)c1Cl N1(C(C(C=C)(F)F)=O)CC(C2CCN(C(=O)Cc3cn(C)nc3Cl)CC2)C1 C1(N(c2ncccn2)C(c2ccc(OC)cc2Cl)=O)CCCCC12CCNCC2 N1(C(CSCC)=O)CCCC(C(=O)NCc2ccc(C(F)C(F)(F)F)cc2)CC1 C1(C(=O)NCC(C2CCN(C(C3CCN(C)C3)=O)CC2)C)CCCCC1O CC1CCCC(C)N(C(C2CCOCCN2C(=O)C(c2cnn(C)c2)=O)=O)C1 Cc1cccn2c(C(=O)NC(CNC(c3ccc4c(n3)CCC4)=O)CO)cnc12 C1(NC(C=CC(C)NC(=O)CC2CC=CCC2)=O)CC2CCC(C1)C2O Cc1cc(C(=O)NCCC2CCCCN2C(=O)CCn2ccnn2)c(C)o1 C1(C(N2CCC(C(C)NC(CC=C)=O)CC2)=O)CCC(=O)CC1C C(=O)(C(F)CC(C)(C)NC(=O)OC(C)(C)C)N1CC(CC)C(C)C1C N1(C(CC2CC(OCC)C2)=O)CCC(NC(c2coc(Cl)c2)=O)C1(C)C N1(C(C2N(C(CC(CC)C)=O)CC=C2)=O)Cc2cnn(C)c2C1 c12cccc(c1)C1CC1C(=O)O2.C(=O)(CCCC1CC1)NCCC(CC(C)O)=O C1(CC(=O)NCC(n2cnnc2)C)CCN(C(=O)CCc2ccco2)CC1 c1(C(N2CC(O)(CNC(c3n(CC)ccc3)=O)C2)=O)ccc(OC)c(OC)c1C C(CCN(C)C(c1cccc(CC(C)C)c1)=O)(C(C)C)NC(C(CSC)O)=O N1(C(C2C3CN(C(C4OCCN(CC)C4)=O)CC32)=O)CCC(F)(CO)CC1 Cc1c(NC(=O)CC2C(NC(C3CCC(F)CC3)=O)CC2O)cnn1C(C)C C1(CC)CCC(C(=O)NCC(C)(C)NC(=O)C(CC)N(C)C)CC1 CC(C)C(C(=O)NCCc1ccco1)C(C)NC(=O)CCS(C)(=O)=O C1(C(=O)N(C)CC2CCCCO2)(CC)CC=CC1.C12CC(C1)C(=O)NCC2 N1(C(C(=O)NC(C)C)=O)CCC2(CC1)CCN(C(=O)C(C)(C)n1cncn1)C2 c1(C(=O)NCC(C)CNC(C2CC3CCC2CC3)=O)cc2ccsc2s1 N1(C(CCC(=C)Cl)=O)CC2CC1CN(C(c1cncc(N3CCOCC3)c1)=O)C2 C1(C(N2CCC(C(=O)Nc3cnc(Cl)nc3)(SC)C2)=O)CCC2CC1CO2 C1(COC)(NC(c2ccc(C)nc2Br)=O)CCN(C(c2cnsn2)=O)CC1 CCCCCCCCCC(C)CCNC1CCC(C)C(C)C1 N1(CC(=O)N(CCCCCNC(c2ccncc2)=O)C)C(=O)CC(C)(C)C1=O S(=O)(=O)(c1cccs1)NCCCNc1cc(C)nn1C1CCOC1 C#CCC(C)C(=O)N(C1CCN(C(=O)C=COCC2CCCO2)CC1)CC1CC1 C1(C(N2C(CNC(C(c3ccsc3)C)=O)CN(C)CC2)=O)OCCOC12CCC2 C1(CNC(=O)NCCn2ncc(CC)c2)CCC(C)(CC)O1 c1(CC(C(=O)NC2CC(N(C(=O)CN3CCCC3=O)C)C2)O)ccccc1Cl c1(C(=O)NC2CC3CC(NC(=O)Cc4nc[nH]n4)C2C3)ccc(O)nc1Cl c1(CNC(C2CC23CCN(Cc2cccc(Cl)c2F)C3)=O)cc2ncsc2[nH]1 c1(C2(CNCC3OCC(CSCC)C3)CC2)ccc(Cl)cc1F.n12cc(nn1)C2 c1(CC(=O)NC2CC(CNC(c3c(C(C)C)ccs3)=O)C2)c[nH]c2ncccc12 C12CC3(C1)CC(C3)C(=O)N(CC(C)(C)C)C2.CC1(C)CN(CC(F)(F)F)C1 C1(NC(CC(=C)C)=O)CC(CNC(c2cc(CC)ccn2)=O)C(O)C1 N1(CC(=O)NCC2CC2Nc2ncc([N+](=O)[O-])cn2)Cc2ccccc2C1=O CC1(C(=O)NCCOC2CCN(C(c3csc(O)n3)=O)C2)COC(=O)C1 CC1C(NC(=O)CN2CCCCCC2)CC2CCC1N2C(=O)Cc1cnn(C)n1 n1(C(C)C)ncc(Cl)c1C(=O)NC(C)CCNC(=O)C(C#N)=CC1CC1 C1(C(=O)NC2(CNC(C3C(OCC)C3C)=O)CC2)COCCC1C c1(N2C(=O)CC(C(N3CC(O)C(O)C3O)=O)C2)ccc(Br)cc1F C1(C(C(=O)NC2CCCOC2)N(c2ccccc2C)CC)C2(CCC2)C12CCC2 C(N=c1ccnc(NCc2cc(=O)cc[nH]2)[nH]1)c1ccc(OC)c(F)c1 Cc1cncc(C2(C(=O)NCC3(CCNC(=O)C=CBr)CC3)CC=CC2)c1 CCCC(O)C(=O)NC1CCN(C(=O)Cc2cnn(C)c2)C1C(C)C c1(C(=O)NCC2(F)CCCN(C(c3nc(C)sc3C)=O)C2)nccn2ccnc12 N1(C(c2c(C)occ2)=O)CCC(C)C1CNC(C1CC2CCC1O2)=O C(CC(CNC(=O)CCCc1nc(C)no1)NC(=O)CSC(C)C)OC CN(C)S(=O)(=O)N1CCC(NC(=O)NCC2CCCC2c2nncn2C)CC1 C1(C(N(CCN(CCOC)C(c2cccs2)=O)CC)=O)CCC(C)(C)C1 Cc1csc(=O)n1CC(=O)OCc1ccc(CSc2cccc(O)c2)o1 N1(C(C23CN(C(C=Cc4scc(C)n4)=O)C(C2)CO3)=O)CCC2(CCCOC2)C1 CC(CCC(C)(C)C)NC(=O)C(CC(F)F)N(C(=O)CCc1nccn1C)C C(=O)(N=c1[nH][nH]c2c1CN(C(c1cnc(C)cn1)=O)C2)c1nccc(COC)c1 n1(C(C)C)ccc(C(N2CC(NC(C3CCC(C(C)(C)O)CC3)=O)C2)=O)cc1=O N1(CC(=O)NCC2CCCN2C(=O)C=CC2CC2)CCNC(=O)C1 c1(NC(C(c2ccn(C)c2)C)=O)ccc(CSc2ccccc2)cc1 N1(C(c2cc(C)ns2)=O)CCC(C2CC2)C1C(=O)NCCCC(N)=O C(C(C)C(=O)N(CCC(=O)NC1CC=C(C)CC1)OC)OCCOC CC(Cn1cccn1)C(=O)N(C1(C(=O)NC2(n3cccn3)CCC2)CC1)C CC(=NO)C1CC(C(=O)NC2CN(C(=O)CC3CCCC(=O)N3)CC2C)C1(C)C n1(CC(=O)NC2CCN(C(C(C)(C)n3cc(Cl)cn3)=O)CC2)cc(F)ccc1=O C(=O)(CCC(=O)COC(C12CCC(CC1)CC2)=O)OCC N1(C(=O)NC(CC#C)C(=O)NC)CCC2C(CC)C2C1 c1(CC(N2CC(NC(CC3(OC)CCC3)=O)C(F)C2)=O)ccc(F)cc1Cl c1(NC(CCCNC(C=CC)=O)=O)cnc(OC)c(C)c1 C(=O)(CCC(F)(F)Cn1cc(-c2ccc(F)cc2)nn1)N1C(COC)COCC1 C1(NC(C2C(NC(c3ncn(C)c(=O)c3)=O)CCC2)=O)CCn2nnnc2C1 c1(NC(c2n(C(C(=O)OC)C)nnn2)c2ccsc2C)cc(CO)ccc1C C1(N(C(c2cc(C(=O)OC)oc2C)=O)C)CCCN(C(=O)CCC(C)=O)CC1 C1(CCC)CN(C(c2cc[n+]([O-])cc2)=O)CCN1C(=O)CCC1CC(C)(C)CO1 C1(C(N(CCOCC#C)C)=O)CN(C(=O)C(F)C2CCCC2)CCC1(C)C C(=O)(C(C(C)(C)C)c1ccccc1)NC(C)C(C)(C)NC(=O)Cc1cnn(C)n1 C(=O)(C1=COCCC1)N1CC(CC(N2C(CC)CC(O)C2)=O)C1 N1(CC(=O)NCCNC(C(C)(C)NC(=O)OC(C)(C)C)=O)CCCOC1=O c1(NC(C2C(CNC(c3c(CC)cco3)=O)C2)=O)cc(C)c(F)cc1F C1(NC(C(CSC)OC)=O)CCCC2CN(C(c3ccc4c(c3)OCO4)=O)CC12 C1(CNC(c2c(OC)cccc2F)=O)CCN(C(=O)C(C)O)CC1(F)F N1(C(C2C(n3cc(-c4ccn(CC)n4)nn3)CCCC2)=O)CCC(O)(SC)CC1 C(=O)(C1CCCc2c[nH]nc21)NC1(C)CN(C(c2ncc(C)nc2)=O)C1 CC(C)CCC(=O)NCC(=O)NC1(CCNC(C2C3CC3C3CC23)=O)CCC1 C#Cc1ccc(F)c(C(=O)NC(C2CCCCN2C(c2cc(Br)n[nH]2)=O)C)c1 CCCCCC(O)CC(=O)NC(C1CCCN1C(c1ccc(C)c(C#N)c1)=O)C C(C)(C)(CCC(=O)NC(c1cccc(F)c1)C)NC(C1C(CCOC)C1)=O CC1CCN(C(C2CSC2)=O)CC1CC(=O)NCC(C1CC1)N(C)C c1(CC(N2CC(NC(C(C)CN3CCCCC3)=O)C2)=O)nccc2ccccc12 Cc1cc(=NC(=O)CC2CC3CCC2N(C(=O)OC(C)(C)C)C3)[nH]n1CC(C)C Cc1csc(CC(N2CCCC2C(C)(C)C(=O)NCc2cnc(C)s2)=O)c1 C1(C(=O)NC2CCCSCC2)CCC2(CC2)N1C(C1CCCC1)=O N1(C(Cc2c(OC)cccc2)=O)CCC2(CCC2)C(C(=O)NC(C2CCC2)C)C1 CC(C)(CCNC(=O)CCn1cccc1)NC(=O)CC1CSC1 C1(CC)CCN(C(C2(CNC(C3C4CCCC34)=O)CC2)=O)C1 c1(C(C)NC(CCC(=O)OC)=O)ccc2c(c1)CCN2CCSC(C)C CC(=O)C(C)CC(C)C(=O)N1C2CCC1CN(C(=O)COC1CC=CC1)C2 Cc1cc(CC(=O)NCC(c2ccccc2)CNC(C2CC(C)(C)C2)=O)cs1 C1(C(=O)NC2CSC2)CN(C(C2CN3CCC2CC3)=O)C2(CCC2)C1 N1(C(c2ncc(OC)nc2)=O)CCC(NC(=O)C(F)=CCCF)C(C)(C)C1 c1(OC)ccc(Br)cc1CNc1cn(C)c(C(N2CCC(C(F)(F)F)C2)=O)n1 Cc1cc(OCC(=O)NCC(C)(C)NC(c2c(C)cncc2C)=O)ccc1F C(c1cccc(C#N)c1)=CC(N1CC(C2(NC(C(CC)OC)=O)CC2)C1)=O C1(CNC(C(C=CC)O)=O)CN(C(c2cnc3n2CCOC3)=O)CC12CCC2 C1(C(=O)NC2(c3cn(CCc4ccccc4F)nn3)CCC2)C2CC3C(C2=O)C13 N1(C(C2C(CC)OCC2)=O)CCN(C(c2nnc(O)nc2O)=O)CC1C C1(C(N(CC(C)C#N)C)=O)CC12CCN(C(c1ccnc(O)c1F)=O)C2 N1(C(C=CC=CC)=O)CC2CC2(NC(=O)Nc2cccc(I)c2)C1 N1(C(c2coc3cc(F)ccc23)C(N2CCCCC2)=O)CCC2(CCSCC2)CC1 CCC(Cc1ccccc1)CC(=O)NC(C)CCNC(c1ncnc(O)c1Br)=O N1(C(C(C2CCOC2)OCC)=O)CCC(C(C)NC(=O)CC2CC(C)=NO2)C1 C(=O)(C1CCCn2nccc21)NCCCC(C)NC(c1ccc(C)c(CO)c1)=O C1(NC(C2CCCOC2)=O)CN(C(c2ccc(N3N=CCC3=O)cc2)=O)CC1F C(=O)(C1Cc2ccccc21)N(C1CCCN(C(c2nc(CC)sc2)=O)CC1)C c1(C(C)=O)ccc(C(=O)NC2CC2CNC(=O)C(Cl)=CCl)cc1F C1(NC(C2CN(CC(=O)C(Cl)(Cl)Cl)C2)=O)CC(O)CN(Cc2ccc(Cl)c(Cl)c2)C1 c1(NC(c2n(C3(C)CC3)nnn2)(C)CC2CCCC2)cc(C(N)=O)c(Cl)c(Cl)c1 Cc1c(C(=O)NCC(C(C)C)NC(C2(O)CCC(C)CC2)=O)cccc1C1CC1 N1(CC(=O)N(C2(C(=O)N3CCC3)CC2)C)CCCCC1=O.C(CCO)CC=CCS c1(CNC(=O)NC2CCOC(C3CCOCC3)C2)cc2cnccc2[nH]1 c1(CNC(=O)C(N2CCCC3(CCCO3)C2)=O)cccc2c1CCS2(=O)=O C#Cc1cc(F)c(C(=O)NC2CC(CNC(C3CC4(C3)CC(O)C4)=O)C2)cc1F C(=O)(CC(C)(C)C1CCCO1)NCC#CC(=O)NCC(=O)N(c1ccccc1)C c1(C(=O)NCC2C(CNC(c3c(C)nsc3)=O)C2)cnn2c(C)ccnc12 c1(C(=O)NC2(CCNC(c3cccc(C(N)=O)c3)=O)CC2)cccn2cncc12 CC1C(NC(=O)C(N2CCCCC2=O)C)CCCN1C(=O)CC12CCC(CC1)C2 C1(C(=O)NC2(COC)CN(C(c3c(SCC)cccn3)=O)C2)CCCC(C)CC1 C(=O)(CC(CC)C(C)(C)C)NC1CC2(C(C(=O)NC(CC#C)CCOC)C2)C1 C(=O)(CN=c1cc[nH]cc1)N1CCCCC(NC(c2cscc2C(F)F)=O)C1 C1(C(N2CCC(n3cnnn3)C2)=O)C2CC(O)C(C2)N1C(C1CCC(=O)O1)=O C(C(C(=O)NCc1cn(C2CC2)cn1)C(C)C)NC(C(CC)(C)C)=O C1(CCNC(C2CC2(Cl)Cl)=O)(NC(C(N2CCSCC2)C)=O)CCOCC1 C1(C(F)(F)F)(C(=O)NCC(C)(C)NC(c2cn(CC)nc2)=O)OC2CCC1C2 c1(C(=O)NCC(C2N(C(CC)=O)CCC2)(C)C)cc(F)c(CC)cc1F CC(C)C(F)(CNC(c1csc(O)n1)=O)C(=O)NCCN(C)C(C)C C(=O)(C(F)CC(C)C)NCCCCCCN(C(C(COCC)(C)C)=O)C Cc1nnccc1C(N1CC=CC(NC(=O)CCc2ccon2)C1)=O C1(CNC(C(CCC)CC)=O)CC2(CO1)CN(C(=O)Cc1ccsn1)C2 C1(C(N(CCNC(C2CC(C(F)(F)F)CO2)=O)CC)=O)CC(=O)NC(=O)C1 C1(CC#C)CN(C(=O)CCN(C(c2c(CO)n[nH]c2C)=O)C(C)C)CCO1 N1(C(C(C(C)O)(F)F)=O)CCC(C2CC2)(NC(c2snc(Cl)c2Cl)=O)C1 C(=O)(CCCC(=O)NC1CN(C(=O)CN(C)C)CCC1c1ccccc1)N(C)C C(=O)(CN=c1ccnc(Nc2cccnc2)[nH]1)N(CC=C)C(c1ccccc1)C C1(CC(=O)OCC)CCCCN1C(c1n[nH]c(C)c1Cl)C(=O)NC1CC1 N1(C(C(CC)OC2CCCC2)=O)CC(NC(=O)C2=C(Cl)CC2)C2(CC2)C1 CC1(NC(=O)CCCc2ccccn2)CC(NC(c2cc(Cl)c[nH]2)=O)C1 c1(C(N(CCCCCNC(C(n2ncc(C)c2)C)=O)C)=O)cc(C)c(F)cc1Cl CC1OC2(C(=O)NCC3(O)CN(C(C4CC4(C)Br)=O)C3)CCC1CC2 c1(CNC(c2ccco2)CN(C)C)ccnn1C(F)(F)F C(=O)(C(C)(C)C(=O)NCC(=O)O)NCCC1CC(NC(CCOC(C)C)=O)C1 c1(C2C(C(=O)NCC3(CCNC(C4(C(F)F)CC4)=O)CC3)C2)ccccc1 c1(CC)[nH]c(=N)sc1C(N1CCC(N(C(C2CC(F)(F)C2)=O)CC)C1)=O C(=O)(C(C(C)(C)C)NC(N)=O)NCCCN(C(C1(CCCC)CCCCC1)=O)C N1(C(C2C(C)C2)=O)CC2(C1)C(NC(=O)C(F)C1CCOC1)CCS2(=O)=O N1(Cc2cncc(C)c2)CCCC2(CCN(C(=O)Cc3ccncc3)C2)C1 c1(C(c2ccccc2C)C)cccc(Cl)c1.c12cn(nn1)CCO2 c1(OC(c2ccco2)Cc2onc(C(C)CCCO)n2)ccc([N+](=O)[O-])cc1 c1(CN(C(C=Cc2ccc(C3C(C)C3)o2)=O)CCO)ccc(Br)nc1Br c1(C(=O)Nc2scc(C(=O)OCC)n2)cnc2c(-c3ccc(F)nc3)cnn2c1 C1(C(N2C(CCNC(=O)Cn3cccn3)CSCC2)=O)CC2CCC(C1)O2 C1(OC(C(=O)NCC(C2CC2)NC(c2n(CC)nnc2)=O)C)CCCCCC1 Cc1ccc(CNc2ccc(F)c3cnccc23)c2ccccc12 CC1CCC(CNC(c2cc(N)c(Cl)cn2)=O)N(C(c2cc(C(F)F)no2)=O)C1 c1(C(=O)NCCCN(C(C(CC)c2ccccc2)=O)C)ccc(F)c2c1CCC2 N1(C(CCC=CC)=O)CCC(NC(c2noc(C3CC3)c2C)=O)CC1C1CC1 C1(NC(=O)NC(c2ccc([N+](=O)[O-])[nH]2)C)CCc2nnc(C(F)F)n2C1 O=C1COc2ccc(C(N3CCCC(c4n[nH]cc4C(=O)O)C3)=O)cc2N1 C1(NC(CC2CCCC(OC)C2)=O)CC2CCC(C1)N2C(=O)C(C)CS(C)(=O)=O C1(C(=O)NC2(CF)CCN(C(C3(F)CC3)=O)C2)C2CCCCCCC12 CCN=c1cc(-c2noc(N3CCCCCC3)n2)cc[nH]1 C(=O)(C1=CC2(CCOCC2)C1)N1CC(CCNC(c2c(C)cncn2)=O)C(C)C1 c1(C(=O)NC2CCCC(NC(CC(CC)(F)F)=O)C2)cn2c(n1)CC(C)CC2 c1(C(N2CC(CNC(C(N)=O)=O)C(C(F)(F)F)C2)=O)cc2c(cn1)OCCC2 c1(C(=O)NCC2CCC(NC(=O)C(C3CCOCC3)F)C2)n[nH]c2cccnc12 C1(C(N2CC(c3cccnc3)C2)=O)(CNC(=O)C=CCF)CC=CC1 c1(N(C)CC2N(C(Cc3cn(CC)nc3)=O)CCC2)nccnc1C#N CN(CCCC(=O)N(C(C)(C)CNC(C1CN(C2COC2)C1)=O)CCO)N=O N1(C(CNS(NC)(=O)=O)=O)CC2CCCC(N(C)C(C3CSC3)=O)C2C1 Cc1csc(CCC(=O)N(CCCNC(=O)CCC2CCC(C)O2)C(C)C)n1 C(=O)(CC1=CCOCC1)NC(CC)CNC(c1c(C)noc1N)=O C1(C(=O)NCCCC(=O)OC)CC2(CCCC2)CO1 C1(C(N2C(C)(CCC)CC2)=O)CCN(C(C2(OC)CCC2)=O)C(C)(C)C1 N1(C(c2cc(C3(O)COC3)on2)=O)CCOC2(C1)CN(C(C1CC1F)=O)C2 CC1(C)CC(C(N2CC3C(NC(=O)CCn4ccnc4)C3C2)=O)C(C)(C)O1 C1(NC(CC2CCC(=O)C2)=O)CC2CC1CN(C(c1cc(F)c(Cl)cc1F)=O)C2 N1(C(C2C(C(=O)OC)C2(C)C)=O)CCCC(O)(CNC(=O)CC2CC=CC2)CC1 c1(C(=O)NCC2C(CNC(c3n[nH]cc3F)=O)C2)cc2ccc(Br)c(F)c2[nH]1 N1(C(C(N(C)C)C2CC2)=O)CCN(C(C2CCCCC2)=O)C(C(C)(C)C)C1 c1(C(N(C2C(C)CCN(C(C(C)(C)OCC)=O)C2)C)=O)cccc2nc(Cl)cn12 c1(C(=O)NC2C(NC(c3cccc(CC)n3)=O)CCCC2)ccc(F)c(F)c1 N1(C(CCCOCCOC)=O)CCC2CN(C(=O)COC3CC3)CC2C1 C1(N(C)C(c2ccncc2F)=O)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)CC1(C)C C(=O)(CC#Cc1ccccc1)OC(c1ccc(Cl)c(C)c1)CC N1(C(CCc2ccc(C)o2)=O)CC2(CC2)CC1C(N1CCC1C(C)O)=O CCCCC(C)(F)C(=O)NCC1(CNC(=O)CC(C)(C)C(F)F)CCOCC1 C1(C(=O)NC(CCSC)C(=O)NCCCc2cnc[nH]2)CC(=O)NC1(C)C c1(NC(c2scc(NC(=O)OCC)n2)=O)c(SCC)cc(COC)cc1F c1(COCC)nc(N(CCCNC(c2sncc2C)=O)C)cc(C)n1 C(=O)(C1CCc2cccnc21)NC1C2(CCN(C(C(CC=CCC)C)=O)C2)C1 CC1(Cc2cn(CC(=O)NCCc3nccs3)nn2)CCCC1O c1(C(=O)NCC(C)N(C)C(C2CCN(c3ccccn3)CC2)=O)coc(C#N)c1 c1(C2(NC(N3CCC(NS(C)(=O)=O)C3)=O)CCC2)cccc(F)c1 C1(CNC(=O)CC2CCC2)CN2CCCCC2CN1C(c1ccccn1)=O C1(C(N2CCC(N(C(=O)CCN(CC(F)(F)F)C)C)C2)=O)(OCC)CCCC1 C1(CCC=CC)NC(=O)CCN(C(c2ccccc2C)C)C1=O C(=O)(CC(C)CC(C)C)NC1C(C(=O)NC(c2c(OC)n[nH]c2)(C)C)C1 CCC(CCCC(=O)N(CCCO)CCO)NC(C1CCC2CC1CO2)=O c1(C(N(C2CCCCN(C(c3n[nH]cc3F)=O)C2)C)=O)cccn2ccnc12 C12(C(N3CC(C=C)(O)C3)=O)CC(CO)(CN1C(=O)Cc1ccsc1)C2 c1(CC(=O)NC2CCN(C(c3cc(Cl)nnc3O)=O)C2)ccc(F)cc1[N+](=O)[O-] C=CC1(CC(=O)NC(C)CC(C)NC(C2(CO)CCC2)=O)CCCCC1 C(=O)(C(O)CC(F)(F)F)NC1C(C(=O)NC2(C(N)=O)CC2)C2CCC1C2 C(CCC(=O)N1CCCC1CNC(=O)CC1(C)CC1)OC(C)C c1(NC2CCN(Cc3ccc(-c4nc(C)on4)s3)CC2)cnc(C(=O)O)c(F)c1 C1(CNC(C(C)(C)F)=O)CN(C(=O)C(CC#N)c2ccccc2)CC1C(F)(F)F N1(C(c2cnc(C)[nH]2)=O)CC2(CC(NC(C3(CC(F)F)CCC3)=O)CO2)C1 N1(C(c2ccc(OC)nc2)=O)CCN(C(c2ccc(C)c(F)c2)=O)C(C2CC2)C1 CC1=C(C(=O)NCCCC(C)(C)NC(C2CC2C(C)(F)F)=O)SCCO1 C1(C(C(=O)C(c2ccccc2)F)=O)CCCN(C(=O)NC23CSCC2C3)C1 C1(CC)(CNC(c2occc2CNC(=O)C=CCOC)=O)CCCC1 N1(C(C(C)OCC#C)=O)CCCN(C(c2cnc(OC)cn2)=O)CC1C c1(NC(=O)N(C2CCC2)CC2CCOC2)ccc(=O)n(-c2ccccc2)n1 C1(C(=O)NCC(CNC(Cc2cc(C(C)C)no2)=O)C)CCC2(CCOCC2)O1 c1(C(=O)OC)cc([N+](=O)[O-])ccc1S(=O)(=O)N1CC(C#N)C2(CCC2)C1 Cc1nn(C)c2c1C(NC(=O)NCC(C)C1CCC1)CCC2 N1(C(c2ccn3nccc3c2)C(=O)NCCC)c2ccc(F)cc2CC1C c1(CN2CCCC(CC(=O)NCCC3CCCCO3)C2)cc2ncccc2o1 C(=O)(C(C)C(O)C(C)C)NC1CCCCN(C(c2cncc(C)c2C)=O)C1 Cc1nc(N2CCC(NC(c3ccn(C)n3)=O)C(F)C2)nc2ccccc12 CCCC(C)CN(C)C(c1c[nH]nc1CNC(=O)CCc1cnccn1)=O c1(C(N(C2CC(C#N)C2)CC(=O)NC(c2ccccc2)C#C)=O)snnc1C C1(NC(C(n2ccnn2)C)=O)CCC2CN(C(=O)C=Cc3cnn(C)c3)CCC2C1 c1(-c2ccc(F)c(C(=O)OC)c2F)c[nH]c2ccc(NC(=O)CC(F)(F)F)cc12 CC(C)(CNC(c1nc[nH]n1)=O)CC(=O)NC(CO)CC(F)(F)F CN1CCn2ncc(CNC(N3CCC(NC(N)=O)CC3)=O)c21 c1(C(N(C2CCC(NC(CCC(=O)NC)=O)C2)C)=O)cc(F)cnc1O Cc1cc(C(N2CCCC(CN(C)C(c3ncsc3C)=O)C2)=O)c(C)cc1Br c1(C(=O)NCCOCCNC(c2n(C)nc(O)c2)=O)ccc(C#N)c(O)c1 C1(NC(c2ccc(C(F)(F)CF)cc2)=O)C2CC(CN(C(=O)CO)C2)C1CO C1(O)(CC(C2(O)CCSC2)C2CC2)CCCOC1.n12cc(nn1)CNC(=O)C2 c1(C(C)NC(C2(OC)CN(C(=O)Cc3ccc(C)o3)C2)=O)nccc(O)n1 C1(NC(=O)CCSCC(N2CCCC2)=O)CCCN(C(C2CC3(CC3)CO2)=O)CC1 C(C(CO)CC(C)C)NC(C(CCC1CC1)NC(C=CC(CC)C)=O)=O Cc1nc(C)c(C(N2CCN(C(C3CCN(C(=O)C(C)CO)CC3)=O)CC2)=O)o1 C1(CNC(C(C)C2CCCC2)=O)(NC(c2cnco2)=O)CCOCC1 c1(C(N2CCC(NC(CS(=O)(=O)NC)=O)C3(C2)CC3)=O)c(F)ccc2c1OCC2 N1(c2c(C)cc(F)cc2)C(=S)NC(c2cscn2)C2=C1CC1(CCOCC1)NC2=O c1(N(C)C)cnc(C(=O)NC2CN(C(c3ccc(CO)cc3)=O)C3CC23)cn1 c1(C(N2C(CCNC(C(C(C)C)O)=O)CC(F)(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl CCCCC(CCC)NC(=O)CCC(C)NC(=O)CCc1nncn1C c1(C(=O)NC2C(C)CN(C(c3cnc(C(N)=O)s3)=O)CC2)cc2c(o1)CCCC2 N1(c2snc(C(C)(C)C)n2)CCC(C)(NC(C2CC(n3ccnc3)C2)=O)C1 N1(C(c2c(C)c(N)ccc2)=O)CC2CC(NC(=O)C(C)n3cnnn3)CC2C1 Cc1ccc2sc(CNC(N3CCN(C4CCN(C)C4)CC3)=O)nc2c1C C1(NC(C(C)(C)C2CCN(C(=O)COC3CCCC3)C2)=O)CCCC(CO)CC1 N1(Cc2c(C)n(C)nc2)CCC(F)(F)C(C(=O)Nc2cnc(Cl)c(C(N)=O)c2)C1 c1(C(=O)NC2(C)CCN(C(C(CCO)N(C)C)=O)C2)cc2ccc(F)cc2o1 C12(C(=O)OC)CCCC(C(=O)OCc3cn(C)c(=O)n3C)C1C2 CS(=O)(=O)C(CNC(=O)CN1CCCC1=O)CNC(C1C=CCS1)=O C1(O)(CN(C)C(C2CC2F)=O)CCN(C(c2cncn2-c2ccccc2)=O)C1 C(C(C)C(C)C(=O)NC1CCC1CNC(c1cscc1C)=O)OC N1(C(CC23CCC(C)(OC2)C3)=O)CCC(NC(c2ncccn2)=O)C(F)(F)CC1 c1(C(=O)NC(CC(C)NC(c2ccn(C(F)(F)F)n2)=O)C)ccc(F)c(Cl)c1 c1(OC)ccc(CC(=O)NCC(C(=O)O)C2CCOC2)c(Br)c1 C(C)(CCC(=O)N(C)CC1COCCN1C(c1occc1Cl)=O)OCC N1(C(CC(C)(C)NC(C(C)N(CC)CC)=O)=O)CC2(CCC(=O)NC2)C1 C1(NC(CN(CC(=O)OC(C)C)C)=O)CCN(C(=O)CCNS(C)(=O)=O)CC1O N1(C(CC=C)=O)CC(CC=C)(NC(=O)C(C)Oc2ccncc2)C1.C1(C)C(=O)N1 C(=O)(CC(C)CC(C)(C)C)NC1CCC(N(C(=O)C=CCc2cccs2)C)CC1 C1(C(=O)N(CCCCCO)CCO)C2CC(O)C(C2)N1C(=O)COCC1CCOC1 c1(C(=O)NCC(CC)NC(c2cnc(S)nc2)=O)cc2cccc(Cl)c2s1 c1(OC)ncccc1C1CCN(C(=O)Cn2cc(C3(CC#N)CC3)nn2)C1 c1(CNC(C2C(C)C2)=O)nnn(C)c1C(=O)NCCn1cncn1 CCC(CC)(CC)NC(=O)C(C1CCN(C(=O)CCC(C)SC)C1)F c1(OC)cc(NC(=O)C(N2CC3CCN(C(C)=O)CC3C2)=O)cc2cccnc12 C(=O)(N=c1cc(C)n(C)[nH]1)C1CCCC(NC(c2ccc(C)cn2)=O)C1 C1(O)(CC(=O)NC(CC#CC)C)CCN(C(=O)OC(C)(C)C)CC1 CN=c1cc(C(N2CCOC(CNC(=O)CC3CCOC3)C2)=O)cc[nH]1 C#CC1(C(=O)NCC2CN(C(=O)C(C)=C(C)C)CC2C(F)(F)F)CCCCC1 Cc1c(Cl)ccc(C(N2CCC(CNC(C3CNC(=O)N3)=O)CC2)=O)c1Cl c1(C(N2C(CCNC(C(C=C)(C)CC)=O)CCCC2)=O)ccnc2c1ncn2C Cc1cc(C2CC2)ccc1Cl.C12(CCCCC1)C(c1ccccc1)NC(=O)N2 CCC(CC)C(O)CNC(C1(n2cc(C(C)(C)NC(=O)C3CC3)nn2)CC1)=O c1(OC)ccc(C(=O)N(C)CC2CCC(C(C)(C)C)O2)c(F)n1 CCC(CC(=O)NCC(C)NC(=O)CN1CCCCC1)OC(=O)Nc1ccccc1 C(=O)(C1=CCCC1C)NC(C(=O)Nc1c(C)ccnc1)(C)C1CCC1 c1(NCC(C)OC)ncnc(NC2CC(=O)N(C)C2)c1C c1(SCCC(C)=O)ccc(C(N2CCOCC2c2nncn2C)=O)cc1 Cc1cc(F)sc1C(=O)NCC(O)CNC(=O)CCc1ccncc1Br N1(Cc2c(C)cccc2)CCC2C1CCCN2C(c1cnn(C(C)(C)C)c1)=O N1(c2nnc(C)s2)CCC(C(C)N(c2ccccc2)C)CC1 C1(CC(=O)NC2CCC(N(C)C)O2)CN(Cc2noc(C3CC3)n2)CCO1 CCC(CN(C)C)C(=O)NCC(CC)NC(=O)C(c1ccncc1C)C n1(C(c2ccc(O)cc2)C)cc(C2NC(=O)Nc3c(C(=O)O)cccc32)cn1 O=C(CC(C(F)F)n1cccn1)NCCC12CC(CO1)C2 C(C)(CC(=O)NCC1CCN(C(=O)CCF)C1(C)C)(C(F)(F)F)N(C)C C12(C(=O)NCCC(C(C)C)C)CC(CO1)N(C(=O)CC13CCCC1C3)C2 c1(CNC(=O)CNC(=O)CC2(NCc3ccccc3)CCC2)ccc(O)cc1Cl c1(C(C)(C)C)ccc(O)c(C(=O)NC2CC2C(=O)NCCCc2ccccc2)c1 N1(C(C2(CSC)CCC2)=O)CCC(NC(c2cc(Cl)ns2)=O)C(O)C1 c1(C(=O)NC2CC(CCNC(C3(C(F)(F)F)CC3)=O)C2)cccn1-c1nccs1 N1(C(C2N(C(CN(c3ccccc3)C)=O)CCOC2)=O)CCC12CCCOCC2 C1(CC=C)(NC(C2CCC(CO)C2)=O)CCN(C(=O)C(O)CC)C1 N1(C(CCc2c(C)nn(C)c2)=O)CCOCC(CNC(=O)C(C)CN(C)C)C1 C1(C(=O)NC2CC(=O)N(C3CN(c4ccncn4)C3)C2)CCCC(CF)C1 CC(C)CC(C)C(=O)N1CCC(F)(CNC(=O)C(C)(C)C2CCCO2)CC1 C12(C(N(CCNC(c3noc(CC)c3C)=O)C3CC3)=O)CCOC1CS(=O)(=O)C2 Cc1cc(C(=O)NC2CC(n3cc(CSc4nc(C(=O)O)co4)nn3)C2)co1 C(=O)(C1CSc2ccccc21)NC(CNC(c1c(C)c(O)ccc1)=O)C1CC1 C(=O)(CCCCC(C)(C)C)N1CC(OC)N(C(=O)CCOC)CC1 c1(CC(=O)NC2CCC(NC(C(F)OC)=O)C2)cn(C)c2ccccc12 c1(C(=O)NC2CCC(CNC(C3(OC)CCC3)=O)C2)ccccc1OC(C)C c1(NC2(CCNC(C3N(S(C)(=O)=O)CC3)=O)CCCC2)cc(O)nc(O)n1 c1(OC)c(C(N2CC=CC2CNC(c2nc(Br)sc2C)=O)=O)c(C)nn1C c1(OC)ccc2cc(-c3c[nH]nc3C(=O)Nc3cn(C)cn3)ccc2c1 C1(OC)CCCCN(N2C(C=O)CNC(=O)C2)C1.C1(C=O)COCOC1 N1(C(CC2(C)CCCCC2)=O)CCN(C(c2cc[nH]n2)=O)CC12CC2 Cc1cc(C(=O)NCC2CCCN(C(c3nc(O)sc3C)=O)C2)ncc1C(N)=O C(=O)(CCCCCS(N)(=O)=O)NCCCCC(CO)NC(C1(COC)CC1)=O c1(COC2CCN(C(C(CC)N3CCOCC3)=O)C2)cccc(C)c1F N1(C(C2N(C)CCC2)=O)CCC2(CC2NC(=O)CC2CCCCO2)C1 C1(NC(C2CCCN(CC3CC(F)(F)C(=O)N3)C2)=O)COC2(CCCC2)C1 C12(CNC(C3OCC(C)C3)=O)CC(CN1C(=O)CCc1ccc(Br)s1)C2 c1(NC2c3c(cc(C)c(Cl)c3)OC2)[nH]c(=NC(C)C2CSC2)nc2sccc12 CC1=C(C(=O)OCC2CN3CCCC2C3)SCCO1 c1(C(=O)O)ccc(CCc2nc(CN(C(=O)C(F)(F)CO)CCCl)n[nH]2)cc1 CCC(CCC(=O)N(C)CCc1nccs1)NC(C1CC2(CCCO2)C1)=O c1(C(=O)NCC2=CCN(C(C(COC)NC(C)=O)=O)CC2)cccn2ccnc12 C1(C(N)=O)(NC(C(C)(C)C2CCCN2C(c2cnco2)=O)=O)CCOCC1 C1(C(N2CC(N(C(CC(C=C)(C)C)=O)C)C(O)C2)=O)CCc2nc(C)cn2C1 c1(C(N2CCC(C(C)NC(Cc3cnc(C)[nH]3)=O)C2)=O)n[nH]c(C)c1Cl c1(-c2nc(-c3n(CCCOC)ncc3)on2)cc2cc(F)c(F)cc2[nH]1 C(=O)(CC(C)C(F)F)NCC(Cc1ccccc1)NC(C1C(CC)C1)=O C1(CNC(Cn2c(C)nnn2)=O)COCCN(C(C2(CF)CC2)=O)C1 c1(C(=O)NC(C(=O)NCC(C)(C)C2CCC2)Cn2cncn2)cc2n(n1)CCC2 N1(C(C(C)n2cccn2)=O)CC(C(N2CCOC(C)(C)C2)=O)CC1(C)C CN1C(=O)OCC12CCN(Cc1nn(C)cc1S(N)(=O)=O)C2 c1(C(N(C)CC2N(C(c3nn(CC)nc3C)=O)CCCC2)=O)cc(Cl)ncc1N C(=O)(N=c1[nH]ccc2cc(Cl)ccc12)C1C(Nc2ccc(C#N)c(F)c2)C1 C1(O)(C(=O)OC)CCN(C(C2COC(C)C2)C(=O)NC2CCC2)CC1 N1(C(c2c(C)cco2)=O)CCCC(CC(N2CCCC(C(F)F)C2)=O)CC1 C1(NC(C2CCN(C(CC)=O)C2)=O)CC2CC(C1)N(C(c1ccc(=O)oc1)=O)C2 C1(NC(=O)CCCF)COC2(CCN(C(=O)NCc3ccccn3)CC2)C1 Cc1ccncc1NC(C1(N(C(=O)CNC(C2CC2C)=O)C2CC2)CCC1)=O C(CCC1CC1)(C(=O)NOCCCCC1CCCO1)NC(c1ccc(C#N)s1)=O N1(C(c2cc(OC)ncc2)=O)CC2CN(C(c3cc(O)no3)=O)C2C1 C(=O)(N=c1ccn(CCCCC#N)[nH]1)N1CCC(=C)CC1 N1(C(COCCCC)=O)CCC(O)(C(=O)NCCN2C(=O)CCC2=O)CC1 C(=O)(CCCCCCCCCC)N1CCCC(CC(=O)NC(CC#C)CO)C1 c1(C(=O)NCC(CN(C(CCCc2nnc(C)n2C)=O)C)C)cccc(=O)n1C N1(C(C(C)OCCOC)=O)CC(N=[N+]=[N-])CC1C(=O)Nc1cnn(C(F)F)c1 C1(NC(CS(C)(=O)=O)=O)CN(Cc2ccc(C(C)(C)C)nc2)CC1(F)F C1(C#N)(C(=O)NCc2cccc(C(=O)NCCS(CC)=O)n2)CCCCC1 O(NC(=O)C(C)C(C)NC(c1c(C)ncnc1C)=O)CCCC c1(C(N2CC(CCNC(c3cc(CC)no3)=O)OCC2)=O)cc(C)c(F)cc1Cl CC1(C)CCN(C(c2cc(Cl)ncc2O)=O)CC1CNC(c1csnn1)=O c1(CNC(CC(C)C)=O)ccc(CN(C(c2cc(-c3ccns3)on2)=O)CC)cc1 c1(C2CC(C(N3CCC3Cn3cc(CC4CCC4)nn3)=O)C2)ccncc1F C(CC)(C(=O)NCc1csc(C(=O)NC(C)Cc2ccncc2)c1)OCC Cc1cc(=NC(=O)C(=O)N2CC3CC(NC(c4ccc(C(N)=O)nc4)=O)C3C2)[nH]o1 N1(C(C2C(C)OCC2)=O)CCC2(CC1)CN(C(C1CC3(CCCC3)C1)=O)C2 c1(C(=O)NCC(CO)NC(C(=Cc2ccncc2)C)=O)cc(Cl)c(C)cn1 C=CC(CC)CC(=O)N1CC(C)(CCC(=O)NC2(CO)CC(C)C2)C1 C1(NC(CCC=CCC=C)=O)CCCC(CC(=O)N(C(CC)CO)C)C1 CCC(C(=O)N(C(C)CO)CC)NC(=O)COc1ccccc1 CCCCC(CNC(=O)COC1(C)CCC1)NC(=O)CN(C1CCCC1)C C1(C(=O)NCC(C(C)(C)C)NC(C2C(CC)OCC2)=O)CS(=O)(=O)CC(=O)N1 c1(CC)cc(C(=O)NC(CNC(C2CCSCC2)=O)(CC)CC)nn1C c1(C(=O)NC(C(C)NC(CC(C=C)CC)=O)(C)C)cc(F)c(OC)c(Cl)c1 C1(NC(c2cccnn2)=O)CC2CCC1N2C(c1cccc(-n2ccnn2)c1)=O C1(OC)CCCC1C(=O)NCCSCCC(F)(F)F.C12(CC1)CC(=O)NC2 N1(C(C(C)SCc2cccc(C)c2)=O)CC(NC(=O)C(C)(C)C)CC12CCC2 n1(CC(=O)NC(CC)CNC(c2snc(Cl)c2Cl)=O)nc(C)c(Cl)c1C C=CC(C)(O)C(=O)N1CCC(C2CCCCN2C(C23CC(CO2)C3)=O)C1 C(=O)(C#CC1CCOC1)n1cc(C2N(C(c3c(C)oc(C#N)c3)=O)CCC2C)nn1 C1(CCC(=O)NCC(C)N(C(=O)CSC2CCC2)CCOC)CCC(=O)N1 CC1CCCC=C1C(=O)N1CCOCC(C(N2CCC(F)(F)C(F)C2)=O)C1 Cc1nc(C(c2nnnn2C2(C)CC2)NCC2(C)CSC2)cs1 C12(C(=O)NCC(CNC(c3[nH]cc(C)c3)=O)(C)O)CC3CC(C(=O)N1)C2C3 Cc1cn2c(CC(N3CCN(CC(=O)NCC(C)(C)C4CC4)CC3)=O)csc2n1 C1(C(=O)Nc2cccc(NC)c2)(NC(=O)CC(C)(O)COC)CCCC1C C1(NC(C(c2cccc(OCC)c2)(C)C)=O)CCN(C(=O)CCCF)CC1F c1(C(C)C)ccc(C(=O)NCCCN(C(C2CNC(=O)C2)=O)Cc2ccccc2)o1 C1(CNC(C2(C(F)(F)F)CC(=C)C2)=O)CN(C(C2CC2(F)F)=O)CC(C)(C)C1 N1(C(c2nc(OCC)oc2)=O)CCC(CO)(NC(=O)CCCC2CCCO2)C1 N1(C(c2cccc(OC)c2OC)C(=O)NC2CC2)CC(C)OC2(CCOCC2)C1 C(=O)(C(C)(CC)CCC(C)C)NC1CCN(C(C=C(CC)C)=O)CC1 N1(C(=O)CSCC(F)(F)F)CCC(C2CCCN(C(C3CC(=O)NC3=O)=O)C2)C1 C12(NC(C(C)NC(CC)=O)=O)CCC(CN(C(=O)C=CC3CCCCC3)C1)C2 C1(C(=O)NCC2(CC(=O)OC)CCOC2)CC(O)(C2CCNCC2)C1 c1(C(N(C)CC2CC(F)CN2C(=O)C(F)CC2CCC2)=O)ccc2cncn2c1 c12nc(cs1)C(=O)N(CC)C2.C(=O)(CCCn1ccc(C(N)=O)n1)NC C(CCC(C)C)(C(=O)NC1(CF)CCN(C(C2(C)CCC2)=O)C1)NC(C)=O N1(C(CN2CC3(CCN(C(C(C)CC(C)(F)F)=O)C3)C2)=O)c2ccccc2CC1C c1(SC)cnn(C)c1C(=O)NC1CC(C)N(C(c2cccc(=O)o2)=O)C1 c1(C(=O)Nc2c(I)ccc(C)c2)cnn2ccc(C3=CCC(O)CC3)cc12 C1(NC(CCOCCN(C(C(c2cnn(C)c2)C)=O)C)=O)CC2CCCC2C1 CCC(C)C(=O)C(=O)N1CC2(CCNC(=O)C(C)SC)CCC1C2 C1(C(N(CCC(C)OC)C)=O)(OC)Cc2ccccc2C1 C(C1CCCCC1)=C(C)C.C123CC(C1)(C2)C(=O)NOC3 c1(C(=O)NCC2CN(C(C3(C(=O)NC)CC3)=O)CCN2C)nnn2c1CSCC2 C1(C(C(=O)NC2(CC)CC2)C)CCCN(C(=O)CN2CCNC2=O)C1 CC(C)(F)C(C)(F)C(=O)NCC1CCCC1NC(c1ccccc1F)=O Cc1nocc1C(=O)NCC(C)C(=O)NCc1nc[nH]n1 n1(CCC)ncc(C(=O)NC2(CNC(=O)CSc3n[nH]c(=N)s3)CCCC2)c1C c1(C(=O)NC(CN(C(C2CCCC(OC)C2)=O)C)(C)C)ccc([N+](=O)[O-])cc1Cl c1(N(c2ccc(Br)c(C)c2O)C(c2c(OC)nccc2)=O)ccc2c(c1)CNCC2 C1(NC(c2cc(C)nnc2)=O)CC2CC(NC(c3cc(C)c(C)o3)=O)CC2C1 CC1(C)CN(C(=O)CCCN2CCCC2)CCC1NC(=O)C=CC1CC1 C=CC1(CC(=O)NC2CC2(C)C(F)F)CN(C(c2ccn(C(F)F)n2)=O)C1 N1(C(c2cncc(SCC)n2)=O)CCN(C(=O)Cc2cccs2)CC12CC2 c1(CC)nocc1C(N1CCC(C(C)C(=O)NCCC(=O)OC(C)C)C1)=O C1(NC(C2CCC(CC)O2)=O)CC2CN(C(c3cc4ncccn4n3)=O)CC2C1 N1(C(c2cccc(OC)c2O)=O)CCCN(C(c2nnc(O)cc2C)=O)CC1C C(=O)(CCCC(=O)NC1CN(C(C2CC(F)(CO)C2)=O)CCC1F)NC(C)C C=C1CCN(C(=O)CCCCCC)C(C(=O)N(C)CCc2ncccn2)C1 C1(C(C)N(C)CC2CCN(C(=O)Cn3cccn3)CC2)CCC(F)(F)CC1 C1(Oc2cc(C)ncn2)CCCCC1C(=O)N(C1CCCC1)CCNC(CC)C CC1CN(C(c2ccc(C(N)=O)nc2)=O)C(C)CN1C(C1CCC(=O)O1)=O Cc1cc(C)c(CN(C)C(c2nnsc2C(F)F)=O)cn1 O=C(CS(=O)(=O)CC1CCCO1)NCC1CCCCN(C(C2(CCF)CC2)=O)C1 N1(C(C(c2cccc(Cl)c2)CC)=O)CCOC(CNC(C2CN(C)CCO2)=O)C1 C1(NC(Cn2nc(C)c(Cl)c2)=O)CCN(C(=O)C=CCF)CC1O c1(C(=O)NCC=CCNC(C(c2ccc(Cl)s2)C)=O)ccccc1C1CC1 CC1(C(N2CCOCC2C(=O)NCC23CC(CN2C)C3)=O)CC2CCC1C2 N1(C(C(C)c2ccsn2)=O)CC2CN(C(=O)C=CBr)CC2C1 CCCCCCCC(=O)N1CCC(NCc2ccc3c(c2)CCO3)C(F)C1 C1(OC)CC2CCC1CC2CNC(N1C2CCC1CN(C)C2)=O C(=O)(CC(C(F)(F)F)NC(c1nocc1C1CC1)=O)N(CC(C)CO)C C(=O)(CCCCC(C)C)N(CC(CC)NC(c1nccnc1C)=O)C c1(C(=O)NC2C(C(=O)NCCn3c(C)cc(C)n3)C2)ccc2c(c1)ncn2C C1(CNC(C=CSC)=O)CCN(C(C2CC(C(N)=O)C2)=O)C1(C)C Cc1c(N(C(=O)C(CNC(c2cnc(=N)[nH]c2)=O)C(C)C)C)cccc1F C(CC(F)(F)F)CCCNC(=O)C(N1CCC(N2CCCCC2)C1)=O Cc1ccc(C(=O)NC2(C)CN(C(C3CCCCC3F)=O)C2)c(F)c1 C1(N(C)C(c2c[nH]nc2CNC(=O)Cc2ccc[nH]2)=O)CCS(=O)(=O)C1 C(=O)(C(CNC(C1CC1[N+](=O)[O-])=O)CC1CCCC1)N(CCCCC=C)C N1(C(CC=C)=O)CCCOC(CNC(c2cc(N3CCOCC3)ncn2)=O)C1 C1(C(=O)O)CCN(C(C2(c3ccccc3-c3cnc(O)c(Cl)c3)CC2)=O)CC1F Cc1cc(C(CNC(=O)N(C)CCC2CCO2)NC(=O)OC(C)(C)C)cc(C)c1 c1(CC)ccnc(C(=O)NCCCCCCNC(c2ccnn2C(F)F)=O)c1 C1(CNC(C=NOC)=O)CC(F)(F)CN1C(C1CCC(C(N)=O)O1)=O S(=O)(=O)(c1cccc(OC(F)F)c1)NC1CCN(C(c2cc(C(=O)O)no2)=O)C1 C1(NC(CCCN(C)C)=O)CCCN(C(C2(F)C3CCCC23)=O)C1 C1(NC(C(CC)N(C)C)=O)CN(C(c2cnc(OC)cn2)=O)CC(F)(F)C1 Cc1ccc(CN(C(C(c2cn(CC(F)(F)F)nn2)NC2CC2)=O)C2CC2)cc1 c1(C(=O)NCC2CCN(C(C(C(COC)C)C)=O)CC2)c(SC)nc(O)nc1C C1(CC)OCCC1N=c1nc2scnc2c(NCC(C)C(F)(F)F)[nH]1 Cc1ncc(S(N)(=O)=O)cc1NC(=O)COC1CNC1.C(=O)(CCC1CC1C)N C1(C(=O)NCC23CC(C)(C2)C3)CC2(CCN(C(c3cc(S(C)(=O)=O)co3)=O)C2)CO1 N1(C(C2(CC)CCC2)=O)CCCC2(NC(=O)CC3CSCCS3)CCCC12 N1(C(C=C(C)C(C)C)=O)CCCOC(CNC(=O)C(c2ccccc2F)C)C1 c1(C(=O)NC(CCC)CNC(C2CC2Cl)=O)cnn2cccc2c1 CCC(CC(=O)N(CC(O)CNC(c1cnn(CCO)c1)=O)C)OC N1(C(c2cc(CSCCOC)on2)=O)CC=CC(NC(=O)C(C)(C)OC)C1 O(N=C1CCCCCC1)CC(N1CC(C(=O)NCc2nc3ccccc3s2)C1)=O c1(C(=O)NCC(C)NC(C(c2ccccc2)OC)=O)cnc2c[nH]nc2c1 c1(C(=O)NCC(C(=O)N(CCC#C)CC)CC2CCCC2)cccc2ccnn12 C1(C)(C(=O)NC(C(=O)OCC)(C)c2ccccc2)CCCCC1 C1(CNC(c2ccc(OC)cn2)=O)CC2CCC1N2C(c1ccc(C)nc1Cl)=O C1(C2CCN(C(=O)CC3CCC(NOCP(C)(C)=O)C3)CC2)(NC(C)=O)CC1 N1(C(C2(C(=O)OC)CC2)=O)CC2CC(N3CCC(C#N)C3)C1C2 O=C(C=CS(F)(F)(F)(F)F)NCCC1CC(NC(C2CCCO2)=O)C1 Cc1cnc(C(=O)NC(C)(C)CC(N2CCC(C#N)CC2)=O)c(F)c1 c1(NC(C(=O)NC(c2ccccc2Br)CC)=O)cccc(C=CCl)c1 CC1CC2(CCC2)CN1C(=O)CC1CC1CNC(=O)COc1ccsc1 N1(C(C2(CC)CCC2)=O)CC2CCN(C(c3cncc(Br)c3)=O)C2C1 C1(C2CC2)(CNC(CCCCNC(C)=O)=O)CCN(C(=O)Cn2cc(C)cn2)C1 C1(C(=O)N(C(C)CC(F)(F)F)C)(COC)C=CCN1C(C1SCCS1)=O c1(NC(C2CCC(N(C)C)C2)=O)cc(CNC(=O)CN2CC(CF)C2)n(C)n1 C1(NC(=O)C=CC2CC2)CCN(C(=O)C(c2cccc(F)c2Cl)(F)F)C12CC2 c1(N2CCC(OC)C2)ccc(S(=O)(=O)NCC23CC(CO)(CO2)C3)cc1F CC#CCCC(=O)NC1CN(C(=O)C(c2cnccc2C)(C)C)CC1C N1(C(CC)CC)CC(C(=O)NCCCNC(=O)C(C)Cc2ccnn2C)CC1=O c1(C(=O)NC2(C)CCN(C(c3ccc(CC)nc3)=O)CC2)cc2ccccn2c1 N1(C(CC(CC)O)=O)CC(S(=O)(=O)N2CCN(CCSc3ccncc3)CC2)C1 N1(C(C(N2C(CCN3CCCCC3)CCC2)=O)=O)CC2CCCC1CCC2.CN C1(NC(C2(C#C)CCCC2)=O)CN(C(=O)C(F)C2CC2)CCC1C C(=O)(CCCCC(F)(F)F)NCC1CC(CNC(C2(C#C)CC(=O)C2)=O)OC1 C1(CNC(=O)Cc2ccsn2)CCCCC1NC(c1ccc(N(C)C)cn1)=O C1CCCC(=O)ONC(=O)c2cn1nn2.Cc1noc(-c2ccccc2)n1 C(=O)(C1=COCCO1)N1CC=CC(NC(c2[nH]cc(C(C)(C)C)c2)=O)C1 CC1(C)CC=C(C(=O)NC2CC(CCNC(c3csc(S(N)(=O)=O)c3)=O)C2)CC1 C(=O)(CS(=O)CCCc1ccccc1)NC(C)Cc1ccc(C(F)F)cc1 C(CC(C)C(=O)N(CC(O)CNC(=O)CS(=O)(=O)NC)C)=CCC C1(C(=O)NC(CN(C(=O)CCN2CC=CC2)CC)C)CCN(S(=O)(=O)NC)CC1 N1(C(CSc2nc(C)[nH]n2)=O)CCC2CN(C(=O)CC3CCS(=O)(=O)C3)CCC12 CC(C)C(C#N)C(=O)N(CCNC(c1ocnc1Cc1ccc(F)cc1)=O)C(C)C c1(C(N2C(CNC(C(c3ccccc3)OCC)=O)CC2)=O)cc(F)n(C)n1 CC(CC(=O)N(CC(C)NC(C1(CF)CCC1)=O)C)NC(N)=O C1(CNC(C2(CF)CCN(C(c3nc(=N)[nH]cc3)=O)C2)=O)C2CCCCCC12 C(C(=O)N=c1c(Br)c[nH]cc1Br)C1CC(NCc2ccc(C#N)c(F)c2)C1 n1(C(C)C)ncc(C(=O)NCC2CC(CNC(=O)CCN3CCCC3=O)C2)c1N c1(CC(=O)NC(CC(C)NC(C(C)NC(=O)NC)=O)C)cccc(C(=O)OC)c1 N1(C(C=C(C)C)=O)CCC(CC(=O)NC(c2ccc(C)cc2)C)CC1 c1(C(N(CC(C)NC(c2cnn(C)c2C#N)=O)C)=O)cnc2c[nH]nc2c1 N1(C(C(n2cc(-c3ccc(O)cc3Cl)nn2)C)=O)CC(=O)N2CCCCC2C1 N1(C(=O)NC(C)(C)C)CC2CN(C(=O)Cc3cnn(C4CC4)c3)CC2(C(=O)O)C1 c1(C(N(CCC(=O)NCCc2cnc(C)s2)CC)=O)cc[n+]([O-])cc1 CCC(CC(F)F)C(=O)NC1CC2CN(C(=O)C(C)NC(=O)NC)CC12 c1(C(=O)NC(CC(C)NC(C2CC(CC)(CC)C2)=O)C)c(C)ncn1C C1(CNC(CC(C)O)=O)CN(Cc2c(F)cccc2F)CCC1(F)F C1(CC(=O)NC2CC(C#C)C2)(NC(c2c[nH]ccc2=O)=O)CCCCC1 c1(CCC(N2CCC(C(C)NC(C3CCCC3(C)C)=O)C2)=O)ccc(O)c(F)c1 N1(C(c2c(CC)onc2C)=O)CCCC2(NC(c3cn(C4CC4)cn3)=O)CC2C1 Cc1ccc(C=CC(N2CCC(F)(CNC(=O)Cc3cncn3C)C2)=O)o1 C=C(CNC(c1nc[nH]c1C(C)(C)C)=O)CCNC(C1(C)CCCO1)=O c1(OC)cccc(O)c1C(N1CC2C(CNC(c3conc3C(C)C)=O)C2C1)=O O=C1Cc2c(C(=O)NCC3CCN(C(C4CC5CCC(C4)O5)=O)C3)cccc2N1 C1(C(=O)NC(CNC(c2n(C)nc(C3CC3)c2)=O)CO)Cc2ccccc2CO1 c1(C(N2CCCC(N(C(=O)C=Cc3cncs3)C)C2)=O)cccn2nccc12 c1(C(=O)NC(CC=C)CNC(c2cc(N)cc(O)n2)=O)sc2nnc(S)n2c1C c1(C(C(=O)N(CC(CNC(C2C(COC)C2)=O)C)C)F)ccccc1 Cc1ccc(CN2CCCC(NC(c3ccccc3Cl)=O)CC2)c([N+](=O)[O-])c1 C1(C(=O)OC2CC3(CCCC3)C2)CCC2(CCOCC2)C1 C(=O)(C(O)C(F)(F)F)N1CCCC(C(=O)NCC2CN3CCC2C3)C1 c1(C(N2C(CCNC(C3ON=C(CC)C3)=O)CSCC2)=O)cc2c(s1)CCCC2 C1(C(=O)Nc2cccc(NC(C(C(C)C)F)=O)c2)COc2cc(Cl)ccc2C1 C(=O)(C(O)C1=CCCCC1)NC1C2CN(C(Cc3cn(C)nc3)=O)C1C2 CCCCC(CNC(c1csc(C(C)C)n1)c1nnnn1CC1CCCO1)CC N1(C(c2ccn(CC(C)C)n2)=O)CCCN(C(=O)CC2CC3CC3C2)CC1C C(=O)(C(CC(=O)NC1CCCCC1NC(=O)C(C1CC1)N(C)C)C(C)=O)OC c12cc(ccc1F)NC2=O.CC=O.C(C=CCN(C)C)N CC1CN(C(=O)CCCCn2ccnn2)CCC1NC(=O)CC1CCCCC1 c1(SC)cc(C(=O)N(C(C)CN(C(=O)COCc2cscn2)C)C)oc1C C1(NC(c2c(CC)cco2)=O)CC2COCC(C1)N2C(c1nnsc1N)=O CC(C)CC(C(=O)N(C1CCCCC1NC(=O)CN1CCOCC1=O)C)C(N)=O c1(C(=O)NC2CN(C(CCC#CC)=O)CC2C=C)cc2c(=O)[nH]ccn2n1 Cn1ncc(C(=O)NCCSCc2nnnn2C)c1-n1cccc1 c1(C(=O)NCC(CNC(C2N(CC)CCC2)=O)O)cnnc(O)c1 c1(NC(C2CC(F)CN2Cc2cc3ncccc3o2)=O)cnccc1[N+](=O)[O-] CC(=O)CCCC(=O)NC(C)(C)CNC(c1ccnc(Cl)c1N)=O CC(=O)CC(C)(C)C(=O)NC1COCCC1C(=O)NC(C)CN(C)C(C)C N1(C(C2CC(C)C2)=O)Cc2ccccc2C(NC(=O)Cn2ccc(O)nc2=O)C1 C1(C(N2CC(C)(NC(=O)C=Cc3cncnc3O)C2)=O)CC2CCCCC2O1 c1(C(=O)NCC(CCl)NC(c2ccc([N+](=O)[O-])o2)=O)cn2c(n1)CCC2 c1(CC)[nH]nc(C(=O)NCCC2(O)CN(C(=O)C(=Cc3cccs3)C)C2)c1C C1(NC(=O)C=Cc2cncc(F)c2)CC2CN(C(=O)C3=CCCC3)CC2C1 c1(OC)ccc(CNC(=O)C(C2CCCC2)Nc2cn(C)cn2)cc1 c1(C(=O)NCCC(=O)OC)ccc(CCNC(C2CCCC2SC)=O)cn1 CC(C)(CNC(C1COCOC1)=O)C(=O)NCC12CC(CCO1)C2 C12(NC(c3cc(C)c(C)o3)=O)CCCC1CN(C(c1ccc(=O)n(C)n1)=O)C2 N1(C(C2ON=C(C)C2C)=O)CCC(CNC(C2(N(C)C)CC2)=O)C(F)(F)CC1 Cc1cc(F)c(C(=O)NCC2(NC(c3c(C)nsc3Br)=O)CC2)cc1F C12(NC(c3cnns3)=O)CCC1C(=O)N2.C1(OC)CC(OCC)C1.C(CO)O CCCCC(CC)CC(=O)NCC1CC(O)CN1C(c1cc(F)cc(F)c1F)=O C1(NC(CC(c2scc(C)c2)O)=O)CCC2(CC1)CN(C(c1cocn1)=O)C2 CCC(C(=O)NCC(C)(C)NC(c1ccc(Cn2cncn2)cc1)=O)C(C)C N1(CC(=O)N(C)CC2(NC(C3CCS3(=O)=O)=O)CC2)CC(=O)NC1=O C(=O)(C1CCCn2nccc21)NC1C(NC(CCCN(C)C)=O)CCC1 CC1(C)CN(C(c2cccc(I)c2)C(=O)O)c2ccc(C(F)(F)F)cc21 c1(C(=O)NCC2(F)CC(NC(=O)C(=O)Nc3ccccc3O)C2)ccccc1O C12N(CCC1(C)C)CCC1CC1CNC(=O)C2.C12CC1N2.C(C)(C)(C)OC C(c1ccncn1)=CC(=O)NC(C1(O)CN(C(c2ccnn2CC2CC2)=O)C1)C N1(C(Cn2c(C)csc2=O)=O)CCC(NC(c2cc(Cl)cs2)=O)C(O)C1 c1(NC(CC(=O)NC)C2CC2)nc(-c2ccccc2)nc(=NCc2ccco2)[nH]1 CC1(F)CCN(CCC(=O)NCC2CC(Cn3cc(CCO)nn3)C2)C1 C1(CC)CN(C(c2cc(C)n(C)n2)=O)C12CCC2 CC1(C)CCCCC1CC(N1CCC(NC(=O)C2=CCC2)C12CC2)=O C1(C(=O)NCC2(C)N(C(C=C(CCC)C)=O)CC(OC)C2)CCC2CC1C2(C)C c1(NC(CCCC#CC)=O)c2c(nn1CCO)CCC2 Cc1c(Br)noc1C(=O)NC1CN(C(C2OCCC2C)=O)CC1F Cc1sc(C(=O)NCC2(C(F)F)CCN(C(C3(C)CC=CCC3)=O)C2)c(C)c1C CCC(C)(CC)C(c1nnnn1C1CC(C(=O)OC)C1)NCC1(C)CS(=O)(=O)C1 C(C(C(F)(F)F)N1CCN(C(c2cnc(Cl)s2)=O)CC1)NC(C1CC=CCC1)=O N1(C(c2c(C)cc(F)s2)=O)CCCCC1C1CCCN1C(=O)Cc1ccoc1 CC1(C)CN(C(c2n[nH]c(=N)[nH]2)=O)CCC1C(=O)NCC1CCC(F)(F)C1 N1(C(CN(C)C(c2ccc(F)cc2)=O)=O)CC(NC(c2ccoc2)=O)C2(CCC2)C1 c1(C2N(C(C3C(C(N)=O)C3)=O)CCC2)ccc(Cl)cc1Br CCCC(C)(O)CC(=O)N1CCN(C(n2c(=O)[nH][nH]c2=O)=O)C(c2cn[nH]c2)C1 Cc1c(C(=O)NC(C)CNC(=O)CCc2ccoc2)[nH]c2c(Cl)cccc12 Cn1nc(C(=O)NC2CCCC2NC(=O)CC2(C)CC2(Cl)Cl)cc1Cl N1(CC(C)C)CCCC(C(=O)NC(C)CCN(C(=O)C(F)=CC2CC2)C)C1 C1(C(=O)NC(C(C)C)CO)CC12CCN(S(=O)(=O)c1ccccc1)CC2 N1(C(C2CC(OC(C)(C)C)C2)=O)CCC(CNC(=O)CCC(=O)N(C)C)C1(C)C C(=O)(CC(C)(C(F)(F)F)N(C)C)NC(CNC(C=CC(C)C)=O)(C)C1CC1 C(=O)(CC(C)(C)F)NCC(C)NC(c1c(SC)csc1)=O N1(C(c2nc(-c3cn(C)nc3)oc2)=O)CCC(C)(CNc2cnccn2)C1 C(=O)(C(Cc1ccco1)NC(=O)C=C(C)C(C)C)N(C(CC)CO)C N1(C(c2ccc(C)o2)C(=O)N(CC)Cc2cccs2)CCN(CCS(C)=O)CC1 c1(CN2CC(CS(C)=O)C2)cncn1C1(NC2CC2)CC1 c1(OC)ccc(F)c(C(=O)N(C2CC(NC(=O)CCC(C)O)C2)C)n1 C1(CC)CN(C(=O)C(C)(C)CN(C(=O)CCCC2CCCO2)C)C(C)CO1 c1(N(CC(F)(F)Br)C)nc(N)c2c(ncn2Cc2ccc(Cl)c(F)c2)n1.CC C1(C(N(c2cccnc2)CC)=O)CCC(C)(C)N(C(C2CC(=C3CCC3)C2)=O)C1 Cc1cc(Cl)ncc1CC(N1CCC(NC(=O)C(F)C2CC2)CC1)=O CCCCC(O)CC(=O)NC(C1CCCN1C(c1cc(C)c(Cl)s1)=O)C c1(C(=O)NC23CC(NC(c4[nH]cc(CC)c4)=O)(C2)C3)c(C(N)=O)n[nH]c1C Cc1ccc(C)c2c(C)c(C(=O)NC3CC4CC3N(C(C3CCOC3)=O)C4)oc12 C=CCN=c1[nH]cc(C(=O)NC2CC(CNC(c3c(OC)ccc(F)c3F)=O)C2)s1 N1(C(c2scc(C)c2)=O)CCC(NC(=O)C(C)C(O)CC)C12CCC2 N1(C(COc2ccc(OCC)cc2)=O)CCOCC(NC(=O)C=CCN(C)C)C1 c1(NC(C2CC(F)CN(c3ncncc3I)C2)=O)c(Cl)cc(Br)cc1[N+](=O)[O-] c1(C(N(CCCC(=O)NCC2(CC)CCCC2)C)=O)n[nH]c(C)c1Cl c1(OCC)nccc(C)c1C(=O)N(CCCNC(C1CCC(C)S1)=O)C C1(NC(N(C2(C(N)=O)CN(C(=O)OC(C)(C)C)C2)C)=O)CC2CCCCCC2C1 CC1CCN(c2nc(-c3ccc(Cn4ccnc4)o3)no2)CC1 C12(CC=CC1)C(=O)N(CCCCCC)CC(=O)NC2.c1(CC)nn[nH]n1 c1(SCC(=O)NC2C=CCN(C(CN3CCN(C)CC3)=O)C2)cc(F)ccc1F C1(CCC(=O)NC(C#C)CC)CCN(C(c2c[nH]nc2C(C)C)=O)C1 N1(C(C(C)C)=O)CCC(C(=O)NCC(O)C(C)(C)O)C(C)C1 c1(NCC(n2cccn2)C)ccc(S(=O)(=O)NC(C)CCC(N)=O)cc1Br S(=O)(=O)(c1ccc(=NCC23CCCC(CO2)C3)[nH]c1)N1CCC(C=C)C1 c1(OC)cc(C(N2CC(O)CC2C(=O)Nc2ccc(C(F)F)nc2)=O)cc(F)c1 C1(NC(c2cn(C(F)F)cn2)=O)CCCN(C(c2ncccc2O)=O)C1 c1(C(=O)NCCC(C)CCNC(=O)C=CCO)ccc(Br)cc1Cl C1(C(N2CCC(OCC(=O)NC3CCC(C(=O)NC)CC3)C2)=O)CCC(C)(C)CO1 CC1C(C)N2C(C)CN1C(=O)C2.c1(N(C2COC2)C)ccccc1 S(=O)(=O)(c1ccccc1C1CC1)NCCCCCC(=O)OC C1(C2CC2)(NC(CCc2c(C)cccn2)=O)CCN(C(=O)COCC2CC2)C1 c1(CNC(C(SC)SC)=O)cc(C(=O)NCC2CC2(Cl)Cl)n[nH]1 C(C(=O)NCC1(C)CCCN1C(c1cncc(F)c1)=O)(C(C)(C)C)OC C1(NC(CCN(CC#C)C(C2CC3(CC(=O)C3)C2)=O)=O)CCOC12CCOC2 S(=O)(=O)(c1ccc(F)cc1F)NCCNC(C1(c2ccc(OC)cc2)CC1)=O N1(C(CCCNS(C)(=O)=O)=O)CC2CCC1C(C(=O)NCC1CCCC(F)C1)C2 C(=O)(NNC(=O)C1CC1Cn1ccnc1)NCc1cn(C)nc1 c1(C(N2CC(C(N)=O)(CNC(c3cc(F)cs3)=O)C2)=O)cccc2oc(=N)[nH]c12 N1(C(C2C(C)(C)C(NC(=O)COCc3cccnc3)C2)=O)CCCC2(C1)N=N2 Cc1nn(CC(=O)NC(c2cn(Cc3ccno3)nn2)C)c(C)c1[N+](=O)[O-] C(C(F)(C(=O)NCCC1C=CCC1)C(C)C)NC(C1(C#C)CCCCC1)=O c1(OCC(=O)NC2C=CC(CC(=O)NC3CCSC3)C2)ccc(N)cc1.C1CC1 C#CCCCC(=O)N1CC(CCNC(=O)C(C(C)C)c2cnn(C)c2)C1 Cc1ccsc1C=CC(=O)NCc1cccc(NC(=O)C(C)N(C)C)c1 C#CC(CC(C)C)NC(=O)NC1CCN(CC(=O)O)CC1 c1(C(=O)NCC(C)CN(C(=O)C(C)(O)C2CC2)C)ccccc1S(=O)(=O)N(C)C Cc1ccc(Cl)cc1C(N1CCC2(CC2C(=O)NCCc2ccsc2)C1)=O c1(CN2CCN(C(c3c(C)c[nH]c3)=O)C3C2C3)c(F)ccc(C(=O)O)c1F C(=O)(C1=CCCC1C)N1CCC(CNC(C=CCC)=O)(OC)C1 S(=O)(=O)(c1c[nH]c(C(N2CC(N(C)C(C3CC4C=CC3O4)=O)C2)=O)c1)NCC c1(CN2CC(CNC(c3ccnnc3O)=O)C2)c[nH]c2cc(Cl)ccc12 CCCCC(C)C(C(=O)NC)N1CCC(O)CC1c1ccccc1OC C(=O)(CC1=CCOCC1)NCCOCCCNC(C(CCCC)ON=C(C)C)=O N1(C(C=Cc2c(C)nsc2)=O)CCCCC(NC(=O)C(C)n2cccc2)C1 C1(NC(C2CCC(=C)CC2)=O)CC2CC(C1)N(C(c1cc(O)nn1C)=O)C2 c1(C(=O)NC2CN(C(CCc3ccc(C)o3)=O)CC2(C)C)ccc2ncnn2c1 C1(NC(C2CCN(CC(F)(F)F)C2)=O)(CO)CCN(C(c2cc(Br)n[nH]2)=O)C1 C1(C)(CNC(CSCCN(C)C)=O)CCCN(C(c2cccc(=O)o2)=O)C1 c1(CCC)onc(C)c1C(N1CC(CNC(=O)CC(C)SC)(COC)C1)=O c1(NC(C(N2CCN(C(c3ccc(C)cc3)=O)CC2)C)=O)cncc(Br)c1Cl N1(C(C(CCC)N(C)C)=O)CCN(C(C2OCCCO2)=O)C2COCC12 c1(OC(CC)C(N2CCCN(C(c3cccnn3)=O)CC2)=O)ccc(F)cc1Cl C(=O)(CC(=O)NCCNC(C1CN(C(=O)Cc2ccc(C(=O)OC)s2)C1)=O)NC N1(C(C2C=CCN(C(=O)CCn3cccn3)C2)=O)CCC(C2CCC2)C1 N1(C(CC(N)=O)=O)CCC(F)(F)C(NCc2c(O)cc(O)cc2O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(N2CCSCC2)C)cncc(OC)n1 CCC(C)(C)C(=O)N1CC(CCNC(C2CC(SC)C2)=O)C(C)C1 O=C(C1CCOc2ccc(Cl)cc21)OCC12COC(C1)C2 CC1CN(C(=O)CC(C)(F)F)CC2(CCN(C3CCN(C(=O)C4CC4)CC3)C2)O1 Cc1cc(C(N2CC(NC(C3(C(C)C)CC3)=O)C3CC23)=O)sc1C c1(C(=O)NC(CNC(C(C)Oc2ccc(C)cc2)=O)(C)C2CC2)cc(C#N)[nH]c1C CC1(C)CNC(=O)C1NC(=O)Nc1cccc(OCCC(C)(C)O)n1 CCCC(C(=O)Nc1cccc(C)c1)NC(=O)NC1CCC(C)(CC)C1 C1(C(=O)NC(CCCNC(C2CC(CCC)OCC2)=O)C)CC2CC1C1CC21 C(CCCO)(c1ccccc1)NC(=O)NCC(COC)O C1(NC(C2(C)CC(=C)C2)=O)CCC(CNC(C2CC2C(=O)OC)=O)CC1 S(=O)(=O)(c1cccc(Cl)c1Cl)N1C(C(=O)Nc2ccc(I)c(Cl)n2)CC(O)C1 C1(C(N(CCCCC)CCO)=O)CCC(C)(C)N(C(=O)CC2C(=O)NN=C2C)C1 c1(C(=O)NCC2(F)CN(C(=O)CNc3cccnc3)C2)cc2ccc(O)cc2[nH]1 C(C)(C(C)C=O)NC(COCC#C)=O.C(CN(C)C)(C(=O)NC)N N1(C(c2ccc(N)c(F)n2)=O)CC2CC1CCC2NC(C1CCCC1O)=O CC1CCN(C(c2ccc(Cl)c(F)c2)=O)CC1NC(=O)CN1CCCNC1=O Cc1ccc(NC2CCCC2C(=O)N(CC(O)CN)C)cc1 C1(C(=O)N(C2CCCC2)NC2CC2)Cc2nccn2C1.O=C1CC(C)CN1 C1(c2ccccc2)(C(=O)OCC(=O)C(F)(F)Br)CCCOCC1 c1(C(N2C(CNC(c3c(CC)ocn3)=O)CCC2)=O)cccc(C2(C#N)CC2)c1 c1(CC(=O)NC2CCCCN(C(c3nc(CC)oc3)=O)C2)ccc2c(c1)CCO2 N1(C(C(CC)N(C)C)=O)C2CCCC1CC(NC(=O)CCC(C)O)C2 C1(NC(=O)NCCOCCC#C)CCOC(C(C)C)C1 C1(CCNC(=O)C=CBr)COCCN1C(=O)CS(=O)(=O)NC1CC1 C1(C(=O)NCCOCCC(=O)NC(c2ccccc2)C)CCCC2CC12 S(=O)(=O)(c1cc(Cl)ccc1Cl)NC1C(C(=O)Nc2nc(SC)nc(O)c2)CCC1 c1(C(=O)NCC2C(CNC(c3cc(OC)nn3C)=O)C2)cc2c(ccn2C)s1 N1(C(C2C(C3CN(C(C4(C)CCNC4=O)=O)C3)C2)=O)CC(O)C2(CCCC2)C1 CCCCC(F)C(=O)N1CCCCC(CCC(=O)NC2(C)CC3(CC3)C2)C1 CC(C)(CC(F)F)C(=O)NC1CC2CCC1(C(=O)NCC#CC#CCO)C2 c1(C(N2C(C)(C(N3C(C(=O)OC)CCCC3)=O)CC2)=O)cc(C)ccc1F CC(C)(C(=O)NCC(n1cc(-c2cn[nH]c2)nn1)CN1CCNC1=O)c1cccs1 C1(CNC(C2CC23CCOCC3)=O)CCN(C(C2(CCF)CC2)=O)CCC1(F)F C1(CCNC(C2CCCS2)=O)CN(C(=O)CCC2CCCCO2)CCO1 C1(C)(C(=O)NC(CCN(C(CCc2cnc(C)o2)=O)C)C)CCCCCCC1 N1(C(CCCCOC)=O)CCN(C(=O)C(c2cc(F)cc(F)c2)C)CC(O)C1 c1(C(=O)NC2CN(C(Cc3cnc(C)s3)=O)C(C)CC2)cnc2c(Cl)cccn12 N1(C(CCc2ccnc(C)n2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccn(C)c1)C2 C12(C(=O)NC(CCNC(C=Cc3c(C)ccs3)=O)C)CCC(N(C)C)(CC1)CC2 N(C(=NCCC(C)=O)NCC1CCOC(C)(C)C1)C1CC(SC)C1 C1(CCN(C(=O)C(F)OC(F)(F)F)C)CCN(C(=O)CC2CNC(=O)C2)CC1 N1(C(CCC=C=C)=O)CCC2(CCCN(C(=O)CCOC3CC3)C2)C1 N1(C(C)C)CCCCC1C(N1CCC(C)(NC(c2cnsc2)=O)C1)=O CN1C(=O)CCCC1C(N1CCC(O)C1C(=O)NC1CCC=CCC1)=O CCCCCCCC(=O)N1CCC(C)C(NC(=O)Cc2cc(C)on2)C1 N1(C(C2N(CC)CCC2)=O)CCC2(NC(C3CC4(CCC4)C3)=O)CCCC12 N1(C(C)=O)CCCC12CCN(C(=O)Nc1noc3c1CNCC3)C2 c1(C(=O)NCCC2(O)CN(C(c3cc[nH]c3)=O)C2)ccc(-c2cscn2)cc1 CCCCC(O)C(=O)NCCC1CC(NC(c2ccccc2NC)=O)C1 C1(NC(C(C=C)(C)C)=O)CC2(CCC(CNC(C3(COC)C=CCC3)=O)CC2)C1 N1(C(COC(CC)C)=O)CCN(C(=O)C(c2cccc(F)c2)F)C(CO)C1 CCC(CC(=O)N1CCCCCC1CNC(=O)CCCOC)CC(F)(F)F c1(OC)oc(C)nc1C(N1CCOC(CCNC(=O)C(C)OCC(C)C)C1)=O C1(CNC(CCC#C)=O)CCCCN(C(c2c[nH]c(Br)c2)=O)C1 CCC(C)C(O)C(C)C(=O)NC1CN(C(C2(C)CCC(=O)C2)=O)CC12CC2 C1(NC(C=C(CC)C)=O)CC(C2CCN(C(=O)CCN3CCCC3=O)C2)C1 N1(C(C(C)S(C)(=O)=O)=O)CC2(CCN(C(c3ccc(C4CC4)o3)=O)CC2)C1 C(CCCN=c1[nH]c2c(c(=NC(C)CN3CCCC3)[nH]1)CCC2)=CC c1(CNC(C(c2ccncc2)N(C(=O)CCc2ccoc2)C)=O)nn(C)cc1[N+](=O)[O-] C1(CN(C(CCNC(C)=O)=O)C)CCN(C(=O)CCC2(C)CCC(=O)N2)CC1 N1(C(C2(CC)CC2(F)F)=O)CCC(O)(CN(C(=O)CCSC(F)(F)F)C)C1 CC1(NC(=O)Cc2ccc(F)nc2)CCCCC1C(=O)NCCOCCC1CC1 c1(C(N(CC(C)CNC(=O)CC2CCCO2)C)=O)cc2cccn2c(O)n1 N1(C(C(C)=C(C)C)=O)CC(F)(F)CC1CNC(c1n[nH]cc1C(C)(C)C)=O C1(CC)C(NC(=O)Cc2cscn2)CCCN1C(=O)CSc1ccc(F)cc1F C#CCCC(O)C(=O)N1CC2(C1)CN(C(C1CCN(C)C1=O)=O)C2 N1(C(C=CC(C)(C)C)=O)CC(CO)C2(C1)CN(C(c1ccc(N)c(F)n1)=O)C2 C1(C(N(C)Cc2ncnn2C)=O)CCC2CCC1N2C(=O)Cn1cnnn1 C1(CNC(c2c(C)nc(C)s2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1C C1(NC(c2c(C)nccn2)=O)CC2(NC(=O)Cc3cnsc3)COC1C2 N1(C(C2N(C(CCNC(=O)CO)=O)CC=CC2)=O)C2CCC1CC1(CC1)C2 CCC(CC(F)F)C(=O)N1CC2(CCN2C(C2(C(=O)OC)CC2)=O)C1 N(C1CCCc2ccoc21)C(C(C(C)NC(=O)CC(C)(C)C)(C)C)=O N1(C(CSCC(=O)OC)=O)CCC(O)(CNC(c2cccc(C(N)=O)c2)=O)C1 C(=O)(C1CCCc2nn[nH]c21)N(C(c1ccc(F)cc1)CNC(=O)CNC=O)C N1(C(C(CCO)N(C)C)=O)CC(CNC(=O)CSCCC(F)(F)F)CC12CCC2 C12(CC(=O)OCC(=O)NCCCN(c3ccncc3)C)CCC(CC1)CC2 c1(CCC(=O)NCC2C(CNC(CC3C(C)(C)CC3)=O)C2)ccc(F)cc1Cl C(=O)(C1c2c[nH]nc2CN1C(=O)COCC1CCOC1)NCC(C)(O)CCO N1(C(CC(CC(C)C)C)=O)CCC2(CC1)CC(C)N(C(=O)Cn1nccn1)C2 N1(C(C(C(C)OC)NC(C(CCC)CC)=O)=O)CCN2C(=O)OCC2C1 c1(NC(C2N(C(c3cn(C)nc3)=O)CC(O)C2)=O)cc(CC(=O)O)c(Br)c(Cl)c1 c1(C(=O)NC2C(N(C(c3c(C)n(C)nc3)=O)C)CCCC2)c(C#N)cnn1C CC(C)CCCN=c1[nH]c(N(CC(=O)NCc2ccccc2)C)nc2c1COCC2 C1(CCNC(CS(=O)(=O)NC)=O)CCCN(C(=O)CCc2c(C)noc2Cl)CC1 C1(C(C)NC(CN(CCOC)C)=O)CCCCN1C(c1nocc1C)=O c1(C(=O)NC(C2CN(C(C3CN(CC)C(=O)C3)=O)C2)C)cnc(C2CC2)nc1C Cc1cc(C(N2CCC3C(NC(=O)CCc4ccc(Cl)s4)CC23)=O)cc(O)n1 C1(F)(C(=O)NCC(c2ccccc2F)NC(C)=O)CCC2(CC1)OCCO2 C1(CNC(C=C(COC)C)=O)CC2(CC(NC(c3n[nH]c4c3COC4)=O)C2)C1 C12(NC(C(C)C)CNS(=O)(=O)CC3CC3)CC(c3ccccc3)(C1)C2F C1(C(=O)NCC2N(C(c3ncn(C)c3)=O)CC(F)(F)C2)CN2CCC1(C)CC2 Cc1ccc(C(=O)NC2(C)CC(NC(C3CCCN3C3CCCC3)=O)C2)s1 C1(N(CC(CC=C)OC(C)=O)CCOC)CNCCN1C(c1ccccc1)=O C(=O)(CCCCCCCC1CC1)N1C(CNC(CN(C(C)=O)C)=O)CC1 c1(C(=O)NCC(N2CC(SCC(C)C)C2)=O)cnc2[nH]ncc2c1 CC(CNC(C1CCCCO1)=O)C(=O)N(C1(CF)CC1)C C1(C(=O)NCc2nc(C)c(C)[nH]2)CC2(CCC2)CN1C(c1ccncc1N)=O N1(C(C2CCN(C)C2)=O)CCN(C(C2CCCN2C=O)=O)C2(CCC2)C1 CC(CNc1cccc(Cn2ccnc2)c1)S(N)(=O)=O C12(CNC(C=COCC)=O)CC(CO1)N(C(C1CC(C(C)C)C1(C)C)=O)C2 c1(C(=O)NC2CCN(C(CCCCCC#C)=O)CC2O)n[nH]c2c1CN(C)CC2 C1(NC(c2c(C#C)c[nH]n2)=O)CCCN(C(c2coc(Br)n2)=O)C1C N1(Cc2cccc(C)n2)CC2(CCC(C(=O)Nc3ccc(Br)c([N+](=O)[O-])c3)O2)C1 N1(C(C(CCOOCCO)NC(C2C(OC)CCC2)=O)=O)C2CCC1COC2.O CC1(C)CCC(C(N2CCC(n3ccnn3)C2)=O)(NC(C2COCC2CO)=O)C1 N1(C(C2(SC)CN(C(c3nn(CC)nc3C)=O)C2)=O)CCC(N=[N+]=[N-])C1 c1(CC(=O)NC(CC(C)NC(c2c(C)occ2)=O)C)ccccc1Cl C1C(C(C)C)C(=O)NOCC(=O)N1.c1(OCC)ccc(=N)[nH]c1 C1(c2c(C)n(C)nc2)C(CCNC(N2CCOCC2C2CC2)=O)CCC(=O)N1C n1(CC)nc(C(N2CCCC2(C(=O)N(C)CC)CCc2cnn(C)c2)=O)cc1C c1(NC(C2C(C(C)=O)C2)=O)cc(C(N2CCCC2CC2CC2)=O)ccn1 C1(OC)CN(C)C(C)(C(=O)NCC2CN(C(c3cncc(C(C)(F)F)c3)=O)C2)C1 n1(CC)ncc(C(=O)NC2(C(=O)NCCc3cnn(CCOC)c3)CC2C)n1 c1(C(=O)NCCC(C)N(C(=O)C(C)CO)C)cnn2c1C(=O)NCC2 C1(C(C(=O)NC2CCC2)N(CC)Cc2cccc(Br)c2)C2CCCCCC12 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(c2cccc(=O)o2)=O)C1 C1(C(=O)NCCC(C)CCNC(c2cc(C(N)=O)[nH]n2)=O)COC2(CCC2)C1 C(=O)(CC1=CCCCC1)N1CC(CNC(CCN(C)CCO)=O)C1 Cc1nnccc1C(=O)NCC1CCC(C(=O)Nc2cccnc2)CC1 c1(C(N2CCN(C(CNC(=O)C#CC3CCC3)=O)CC2)=O)cc(F)c(F)c(F)c1 CC1=CCC(C(=O)NCc2nocc2C(=O)NC2CCC(F)CC2)CC1 C(=O)(C#CC1CCCCC1)N1CCC(C(N(CC(F)(F)F)CC)=O)CC1 c1(CNC(C)C(N2CCCC2(C)C[N+](C(c2ccco2)=O)([O-])NC)=O)ccc2nccn2c1 N1(C(Cc2c(C)ncs2)=O)CCC(C)CC1C(=O)NC(C)(C)CCN(C)C c1(C(N2C(CNC(CN(CCCCCC)C)=O)CC2)=O)cccc(N)c1 CC(C)(C)C#CC(=O)N1CCCC1c1cccc(F)c1.C12CCC(C1)C(=O)NC2 c1(C(=O)NCC2(O)CC(NC(c3cc4n(n3)CCC4)=O)C2)ccc([N+](=O)[O-])s1 c1(NC(C2CCN(C(c3cnc(C)[nH]3)=O)C2)=O)ccc(C)c(C)n1 N1(C(C(CCC)O)=O)C2CCC1CC(CNC(=O)CNC(N)=O)C2 c1(C(N(C2CCN(Cc3c(CC)noc3)CC2)C)=O)occ2c1CCC2 N1(C(C=C(CC)C)=O)CCC(CNC(c2cnn3ccccc23)=O)C(F)(F)CC1 C1(NC(c2cnc(C(F)F)s2)=O)CC2CN(C(c3ccccc3Cl)=O)CC2C1 C(=O)(C(C)S(N)(=O)=O)N1CCC(N(CCOC)C(C2C(C(F)F)C2(C)C)=O)CC1 C1(C(C)NC(=O)CCC2CC(NC(=O)C(F)F)C2)CCCCC1 C(=O)(C1=C(Cl)CC1)NCc1cc(C(=O)NC(c2ccccc2O)C)sc1 N1(CC)CCCC(C(=O)NCC2(CNC(=O)C(C)CC3CCC3)CCC2)C1 c1(C(=O)NC23CC(NC(CC)=O)(C2)C3)cc(O)c(F)cc1F N1(C(c2csc3ccccc23)C(=O)NC2CCCC2)CCCC2(CCC(O)C2)C1 c1(C(N2C3C(N(C)C(C4CSCCS4)=O)CC(C3)C2)=O)cccc2c1CCCC2 c1(-c2scc(C(C(=O)NC3(C)CC3)N(C3CCCC3)C)n2)cccc(Br)c1 C(C(CC(C)C)C(=O)NC1CCC(C#N)CC1)NC(CN(C1CC1)CC)=O C(=O)(CC(C)(C)C#N)N(CC(N1C(C(=O)OC)CC1C)=O)C c1(NC(=NCCc2ncc(C)cn2)NC2CCCC2)ccc2c(c1)C(O)CCC2 c1(CC)ccc(N(C2CCCC2)C(=O)COC2CC(NC(=O)COC)C2)c(F)c1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)Cn2cnc3c2CCCC3)CC2(CC2)C1 Cc1nccc(C(=O)NCc2ccccc2CNC(C2CC23CCCC3)=O)n1 C1(NC(C2(CC)CCCCO2)=O)CC2CCC1N2C(c1cc(F)cnc1O)=O c1(C(N2CC(OC)C(NC(=O)Cc3cnns3)C2)=O)cnc(N)c(CO)c1 CCC(CC(=O)N1CCCC1(C(=O)N(C)CCc1cn(C)nn1)CC)C1CCC1 c1(OC)ccnc(C(=O)N(C2CC(NC(=O)CC(C)OC)C2)C)c1C c1(C(=O)NCC(CNC(c2cnc(S)n2C)=O)OC)cn(C)cc1C(F)(F)F c1(OC)cc(C(=O)NCC2=NOC3CN(C(=O)CSC)CC23)ccc1[N+](=O)[O-] C(=O)(CC(C(F)(F)F)NC(=O)CN(C1CCC1)C)N(C)CCC1(N(C)C)CCC1 N1(C(C2(CC=C)CC=CC2)=O)CC(CNC(=O)CCC2CCCCC2)C(C)C1 N12CC3(CCC(CC3)NC(=O)c3cc(cs3)C1=O)C2.c1(COC)ccc(F)cc1 C12(CC(N3C(C)CC(NC(c4n(CC=C)ccn4)=O)C3)=O)CNC(=O)C(C1)C2 N1(C(=O)CCCF)CCc2c(O)nnc(-n3cc(-c4cc(F)nc(F)c4)nn3)c2C1 c12ccccc1CC(=O)N1CCC(C1)C(=O)O2.CC1CCN(C)C1.C(C)(C)(C)O N1(C(CC(CC2CC2)NC(C(C)(C)CC#N)=O)=O)CCOCC2(CCC2)C1 N1(C(CSCC)=O)CC(NC(=O)Cc2nonc2C)CC12CCC2 c12cc(n[nH]1)C(=O)NC2.C1(CC(=O)OC)CCCC1C(=O)N(C(C)C)CC1CC1 c1(C(N2CCC(C(C)NC(c3cc(Cl)on3)=O)C2)=O)cc[nH]c(=N)c1[N+](=O)[O-] C1(CC)CCN(C(c2cc(C)nn2C)=O)C1C(=O)NCC1CN(C2CC2)C(=O)O1 c1(C(=O)OCC)ccc(C(C)OC)cc1NC(c1cnc(Cl)n1C)=O CCCC(C)(C)CC(=O)N(C1CCC(NC(=O)CN(C2CCC2)C)CC1)C Cc1nc(C)n(CCCCC(=O)NC(C)C(C)(O)C(C)C)n1 N(C1CCOc2c(Br)cccc21)C(C1CC2(CCCC2)CO1)=O C12(C)CCCN1C(=O)CC2.C1(N(C(C2CC(=C)C2)=O)CC)COC(C)(C)C1 c1(NC(=O)CC2CCN(CCn3ncc(C)c3)C2)ccc(C#N)cc1 C12(CCNC(c3cc(C(=O)OC)on3)=O)CCC1CN(C(c1ccco1)=O)C2 C12(CNC(C(C(CC)C)O)=O)CCC(CC1)N(C(c1cn3ccnc3s1)=O)C2 O=C(C1OCCc2ccccc21)NCC1CC(NC(c2cccc(F)n2)=O)C1 C=CC(CC)CC(=O)N1CC(C(C(N2CC(F)CC(F)C2)=O)OC)C1 c1(OC)cnc(SC)nc1N1CCCC(C(=O)NC(c2nc[nH]n2)C)C1 C(C(CNC(c1coc(Br)n1)=O)CO)NC(c1cnn(C2CCCC2)c1)=O N1(C(c2nc(-c3c(C)cn(CC)n3)sc2C)=O)CCC2(CCCO2)C1 C(=O)(C1OCCn2ccnc21)N1CCC(NC(CC2(C)CCCO2)=O)(CO)CC1 C1(C(=O)NCCC2CCN(C(CN(C3CC3)CC)=O)C2)CCCCN1C1CC1 CC1(C)CCC1CC(=O)N(C1CCCCC1)CCNC(c1csc(O)n1)=O C12(NC(c3cc(C)nc(O)n3)=O)CCCC1N(C(c1n[nH]c(C)c1F)=O)CCC2 c1(C(=O)NC(C(=O)NC(CCOC)C)C2(C)CC2)ccc(C#N)c(C)n1 C(CO)(CCC(=O)NCCN1CCCOC1=O)NC(=O)OC(C)(C)C C1(C(=O)OC)N(C(=O)CCCc2csc(=N)[nH]2)CC12CCOCC2 C1(CC)CN(C(c2ccc(C#N)cn2)=O)CCC1NC(C12CCC(CC1)C2)=O Cc1cc(C(=O)NC2CN(C(c3cn[nH]c3)=O)C(C)(C)C2)cc(C)n1 Cc1ccc(CC(=O)NC2CC(C)N(C(c3c[nH]nc3C)=O)C2)cc1 C1(CNC(C2=C(C)CCC2)=O)CC2(CO1)CN(C(C1COCC(C)O1)=O)C2 c12cnc(nc1)CNC2.c1(COC)cccc(Oc2ccc(Cl)cc2)c1 c1(C(=O)NC(c2noc(C3CC3)n2)CC)cc2ccncc2c(O)n1 C(=O)(C(F)(F)C(C)(C)O)N1C(C)CC(CC(=O)N(CCC)CC)C1 Cn1cc(C(=O)NCC2CN(C(C3CCC(CO)CC3)=O)C2)c(C2CCOC2)n1 C1(NC(=O)C=CC(=O)NCCC(=O)NC2CC2)CC(CO)C12CCC2 C1(CNC(CC2(C)CC2)=O)CC2CCC1N(C(C1COCCO1)=O)C2 CC1(C)CN(c2nnc(C(F)(F)F)s2)CCC1NC(=O)CC(F)(F)F CC(C)C(CC(=O)N(C)CC1CCN(C(=O)Cn2cnnc2O)C1)C(C)C Cc1nc2ncccc2cc1CCC(=O)NC(C)CNC(C1CCC(C)(C)O1)=O CC1CC1(F)C(=O)NCCCC1(NC(=O)Cn2cnnc2)CC1 c1(CN(Cc2cc(OC)n(C)n2)Cc2cccnc2OC)cc(C)cc(O)c1 C1(C(=O)Nc2ccc(-c3cn(CC)nn3)cn2)CC2CC2CC1C.N1CCC(CO)C1 c1(C(N(C)CC2N(c3cc(OCC)ncn3)CCC2)=O)cccc2nc(O)[nH]c12 C1(NC(C=CC(CC)=CC)=O)CN(C(c2cc(Br)sc2C)=O)CC1OC c1(C(N2CC(O)CC(NC(C=C3CCN(C)C3)=O)C2)=O)c(O)ccc(F)c1F C(=O)(CCCCCF)NC1C(CNC(C23CC(C)(C2)C3)=O)CCCC1 Cc1cc(C(=O)NC23CCC(C(=O)NC4CCCCC4)(CC2)C3)cc(O)c1 c1(C(N2CC(O)(CCNC(C(C3CCOCC3)C)=O)C2)=O)cnc2[nH]nnc2c1 C(C)(C(=O)OC1C=CCC1)(C(=O)NC(C)(C)C)OC.c12csc(n1)CNC2=O C1(CC(=O)NC(CN(C)C(C2CC3CCC3C2)=O)(C)C)CCn2cncc2C1 C12(C(=O)NC(C=C)(C)C)COCC1CN(C(c1cccc(OC)c1)=O)C2 CC1(CNC(c2cc(Cl)c(Br)s2)=O)CCCN1C(c1cc(C#N)c[nH]1)=O C1(NC(C2CCC(C)(C)C2)=O)CC2CCC1N(C(=O)CCNc1ccccn1)C2 C#CCC(CC(F)F)C(=O)NCc1cn(CC(=O)NC2CCC3(CC3)C2)nn1 Cc1cccc(C=CC(N2CC(CNC(c3ccc(OC(C)C)nc3)=O)C2)=O)c1 N1(C(C(C(C)OC)NC(C(C=C)OC)=O)=O)CC2CCC(C1)C(=O)O2 CC1(C)C(NC(=O)C(F)=CC2CC2)CC1CNC(c1coc(C2CCCCC2)n1)=O c12ccnc(c1)C(=O)N2.C1(C)(COC)CC(C(=O)NCCc2n[nH]c(C)n2)C1 CCCC(C)(C)C(=O)N1CCN(C(=O)C(N2CCN(C)CC2)C)C(CC)C1 N1(C(c2n(CC)ncn2)=O)CC(CNC(c2n[nH]cc2OC)=O)CC1C Cc1cccc(Br)c1N.c1(CNC(C2CC2NCCl)=O)ccc(N2CCCCC2)cc1 C1(CC(=O)NCC(C(=O)NC)O)CCCN(C(=O)Cn2nccn2)C1 C1(COC)CN(C(C2CC(=O)N(C)C2)=O)CCN1C(=O)CC1CCCCCC1 Cc1ccc2c(c1C)OCC2NC(C1COC(=O)N1C)=O c1(N2CC(CC(C)NC(CN(C(COC)=O)C)=O)C2)nc2cc(F)ccc2o1 CCC(CNC(C1(CO)COC1)=O)(CC)NC(=O)CNc1nccc(OC)n1 C1(C)(NC(C2N(CC)C(=O)CC2)=O)CCCN(C(=O)Cc2nocc2C)C1 N1(C(CCC(C)C)=O)CCC2(CC1)CCN(C(=O)C(C)C(F)F)CC2 N1(C(C(C(CC)C)O)=O)CCc2ccccc2C1CNC(c1ccon1)=O c1(CC)cccc(C(N2CCC(C(C(=O)NC3(CC4CC4)CC3)F)C2)=O)c1 CCC(Cc1ccccc1)C(=O)NC1CCN(CCNC(C2CC2F)=O)CC1 C=CCC(C)(C)CC(=O)NC1CCSC12CN(C(=O)CCC1(O)CCC1)C2 Cc1nn(CC(N2CCOC(CCNC(=O)C(C)CF)C2)=O)c(=O)o1 C1(C(=O)NC2(C(N)=O)CC2)CCCN(C(c2cccnc2S)=O)C1 N1(C(CC(C)N(C)C)=O)CCC2CCN(c3ncnc4cc(Br)ccc34)CC2C1 C(=O)(CCCCCCc1cc(Cl)sc1Cl)NCC(C(OC)OC)OC Cc1ccc(F)c(OCC(=O)NCC2(O)CCN(C(c3ccc(C#N)s3)=O)C2)c1 c1(C(C(=O)NCCC(C)(C)NC(C2CC3COCC3C2)=O)OC)cc(C)cc(F)c1 CCC(C)C(CC(=O)N1CC2CC(F)CC2C1)NC(=O)C(C)(C)n1ccnn1 Cc1ccsc1CCC(N1CCC(C(C)(C)C(=O)NC2(C)CC2)C1)=O C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(Cn2c(=O)ccc(C)c2)=O)CCC1 C(=O)(C1CCCc2c(O)cccc21)NC1CN(C(CSC2OCC(C)(C)C2)=O)C1 c1(NC(N(CC(N)=O)C)=O)cccc(S(=O)(=O)NC2CC3CCC2O3)c1 CC(C)CC(C)C(=O)NC(C)(CO)C(=O)N(C)CCc1ccccn1 CC(C)(C#CC(=O)N1CCN2CCCC2C1)CNC12CCC(CC1)C2 C1(CNC(CCC(C)SC)=O)CN(C(c2nc(C3CC3)c(C)s2)=O)CC12CCC2 C(=O)(C(O)CCC(C)C)NC1C(NC(c2c(C)csc2)=O)CCCCC1 C1(NC(CC2N(C)CCC2)=O)CCN(C(c2c[nH]ccc2=N)=O)CC(O)C1 CCC(C)(C#N)C(=O)NCC1CCCCC1NC(c1c(C)cnn1C(C)C)=O N1(C(C2C(CC)OCC2)=O)CCC(CO)(CNC(c2ccc(N)cc2Cl)=O)CC1 C1(CCC)(NC(c2cc(Cl)ccn2)=O)CCCN(C(C2(N(C)C)CCCC2)=O)C1 C(CCC)(C(=O)NC(C1(CN(CC=CC(=O)NC)C)CC1)C)=CCC C1(OC)CN(C(c2c[nH]c(C#N)c2)=O)CC1NC(C1(C)CNC(=O)C1)=O C=C=C(C)CC(=O)NC1CC(CNC(c2ccn(-c3cccs3)n2)=O)C1 c1(OC)cc(=O)n(C)cc1C(=O)N(C(CNC(=O)CC(C)(C)C)C1CC1)C N1(C(C(COCC)(C)C)=O)CCC2CC2(C(=O)NCc2ncnn2CC)CC1 N1(C(CC=C)=O)CC(C2CN(C(C3COC(=O)O3)=O)C2)C1 S(=O)(=O)(c1cn(CC)nc1C)N1CC2N(Cc3ccc(CC)s3)C(CC2)C1 N1(C(C(COC)CC(C)C)=O)C2CCCC1CN(C(c1cn[nH]c1)=O)CC2 C(c1ccc([N+](=O)[O-])cc1)=C(C)C(=O)OC(C(C)C)C1CCC1 c1(C(=O)NC2CC(C)N(c3cnc(F)cn3)C2)cnc(O)c2ccsc12 c1(CNC(CC(C)N(C(CCOCCC)=O)C)=O)cnn(CC)c1C S(=O)(=O)(c1ccc(NC2C3CC4CC(C3)CC2C4)c(C#N)c1)NC.C1(C)CCN1 S(=O)(=O)(c1ccc(C)c(C)c1)NCC(=O)NCC(C(C)C)NC(C1CCCC1)=O C(=O)(C(C)(C)C(C)(C)C)N(CCN(C(C1CCC(NC(C)=O)C1)=O)C(C)C)C CCC(C)(C)C(C)CC(=O)N1CC(CN(C(=O)C2=C(Cl)CC2)C)C2(CC2)C1 C12(C(N3CC(C)OC(C4CC4)C3)=O)COCC1CN(C(c1csc(CO)n1)=O)C2 c1(C(=O)NCC(CNC(=O)CCn2cccn2)O)ccnc2ccncc12 Cc1ccc(CN(C(C2CCN(Cc3ccncc3)C2)=O)C)cc1C C1(C)(CNC(CSC)=O)CCCN(C(c2ccc(C(F)(F)F)cc2N)=O)C1 N1(CCC(=O)NCCN(C(COC)=O)C)CCCCC1=O C1(CNC(CC2(O)CC(C)(C)OC2)=O)C2CCCC1N(C(C1CC(=O)C1)=O)C2 C1(Nc2cc(C(=O)OCC)nc(C)n2)CCC2CCN(C(=O)CCS(C)=O)C12 c1(C(N2CCCC(C(C)NC(c3c(C)cncc3)=O)C2)=O)cc(F)c(F)cc1F C1(NC(Cc2cn(CC)nn2)=O)CC(NC(=O)CC2CCCCN2C)C(O)C1 C1(C(=O)NC2(CCCC(=O)NC(COC)C3CC3)CCC2)CC1C1CCCC1 CCCC(O)C(=O)NCCN(C)C(c1nnsc1C)=O C1(CN(C(C2(C#C)CC2)=O)C2CC2)CCN(C(C2CCOC2C)=O)CC1 N1(CC(N2CC(NC(CC(C)F)=O)C(O)C2)=O)CCC(=O)NC1=O C(N=c1ccc([N+](=O)[O-])c[nH]1)C1(CO)CCCN(C(CC(C(C(C)C)C)C)=O)C1 CC1CCN(C(c2cc(C3(C)CC3)on2)=O)CC1CNC(=O)CCC1CC1(Cl)Cl C(CCCCCNC(C12CC1CN(C(=O)CN(C)C(=O)C1CC1)C2)=O)N(C)C CCCCC(=O)NCC(C1CCCC1)NC(=O)CC(C)n1cccn1 C1(CC(=O)NCC(N2CCN(C(C3CC(F)(F)C3)=O)CC2)=O)CCCOCC1 C1(C#N)(C(=O)NCC(C2CCCCC2)NC(c2cn(C3CC3)nn2)=O)CCCO1 c1(C(=O)NCC2C(NC(c3noc(CC)c3C)=O)CC2)cnn2ccncc12 C1(CNC(C(C(C)C)CO)=O)CCN(C(=O)Cc2cc[nH]n2)CCC1(F)F Cc1c(C2CC2C(N2CCC(OC(=O)CCC(=O)O)C2=O)=O)cccc1Br c1(-c2n(-c3ccc(OC)c(OC)c3)nc(C3CCC3)n2)cc(Br)c(F)cc1Cl S(=O)(=O)(c1ccc(NCc2cncc(F)c2)c(Cl)c1)N1CCCCC(SC)C1 n1(CC(=O)NCC(c2cccc(C)c2)NC(C2C=CCC2)=O)nc(C)c(Cl)c1C N1(C(Cc2ccn(CC)n2)=O)CCCCC1C(N1CC(N(CC(C)C#N)C)C1)=O Cn1c(=O)oc2c(C(=O)NC3CC3CNC(C3CCNC(=O)C3)=O)cccc12 CN1CCC(C)(C(N2CCC(OCCNC(c3ccc(N)cc3Cl)=O)C2)=O)CC1 CCCCC(CNC(=O)CCN(C)CC)NC(c1ccncc1C)=O c1(C(C(=O)NC(CC(C)NC(C2C(=C)CC2)=O)C)OC)ccc(C)cc1 N1(C(c2c(CC)n(C)nc2)=O)CCCC(NC(=O)CSC2CC2)C1C C12(C(N3CCC(N(C)CC)C3)=O)CC(CN1C(C1(Cl)CCC1)=O)C2 c1(N(C2CN(C(C(C=C)(C)O)=O)C2)C)nc(Cl)ncc1CC(=O)NC N1(C(CN(CC(C)C)C(C2CC(F)(F)CS2)=O)=O)CCCOC(C2CC2)C1 c1(NC)cc(OC)ncn1.C12(NC(=O)OCC)COC(C(C)NC=O)(C1)C2.CC c1(CC)ccc(-c2nc(CC(n3ccnc3)C)n(CC)n2)nc1 c12c(F)ccc(c1N)O2.n1(CC#C)ccc(C(N2CCC(CNC(C)=O)C2)=O)n1 CP(C)(=O)c1cccc(C(=O)NCC=CCNC(C2CCN3CCCC3C2)=O)c1 Cc1nc(CC(C)C)c(C(=O)NC(C2CN(C(=O)CC3CCCO3)C2)C)s1 C=C(Cl)C(C)(C)C(=O)NCCC(O)CNC(=O)CN(C)C(N)=O Cc1cc(Cl)cc(C(=O)NC2CC(CNC(C3(C)CC3(F)Cl)=O)C2)c1O C1(CC(N2C(CNC(C(C)SC(F)(F)F)=O)CCC2)=O)CCCC(C)(C)O1 CC(C)CC(C(=O)NCC1CCN(C(=O)C(c2cccs2)C)C1)NC(N)=O N1(C(=O)OC(C)(C)C)CC2CN(CC3CC3F)CC(C1)C2(F)F c1(NC(N2CCN(C(c3ccc(SC)[nH]3)=O)CC2)=O)c(C)ccnc1Cl N1(C(C(CC)C(F)(F)F)=O)CC2CCN(C(C3CC4(CCCC4)CO3)=O)CC2C1 CC(=NO)C1CC(C(=O)OCC(c2c[nH]c3c(Cl)nccc23)=O)C1(C)C C(=O)(C(=O)C(C)(C)C)NCC1(F)CC(CNC(C(=Cc2ccccc2)OC)=O)C1 C=CC(CCC)CC(=O)NC1CC1CNC(=O)Cn1nccc1C C1(NC(C2(NC(c3n(C)c(S)nn3)=O)CCSC2)=O)CC2CCCC2C1 c1(OC)nccc(C(=O)NC2CC(O)(CNC(c3ccc(C4CC4)o3)=O)C2)c1F c1(CN(CC(C)OC)C)ccccc1CNC(=O)NC1CCN(C)CC1 c1(C(C(=O)N(C(C)C)CCNC(C2CC2Cl)=O)(F)F)ccc([N+](=O)[O-])cc1 c1(C(N2CC(CN(C(C(COC)C)=O)C)OCC2)=O)ccc(N)c2ncccc12 C(=O)(CCCCCCS(N)(=O)=O)N1CC(C2(NC(C(C)(C)S(C)(=O)=O)=O)CC2)C1 CC(CN=[N+]=[N-])NC(C1OCCC1NC(c1ccc(CO)o1)=O)=O C1(C)(CNC(CNc2ccc(OC)cc2)=O)CCCN(C(C2CCCO2)=O)C1 c1(CN(C(C(C(CC)C)O)=O)C)cnn2c1CN(C(c1cncc(F)c1)=O)CC2 CC1(C)CN(C(=O)Cc2c(O)ncnc2O)CCC1NC(=O)C(=O)C1CC1 c1(OC)ccc([N+](=O)[O-])c(N2CCCC(c3nc(C)c(C)[nH]3)C2)c1F c1(-n2c(NC(CCSc3nc(C)sc3)=O)ccc2)ccc(Br)c(F)c1 N1(C(Cc2c(C)noc2C)=O)CCC(O)C(C(=O)N(CC)Cc2ccccc2)C1 Cc1cc(-c2ccc(C(=O)NCC3CC3NC(c3c[nH]c(=N)s3)=O)cc2)c(C)o1 C1(C(N(C)CCNC(c2cnc3n2CCC3)=O)=O)COc2ccc(Cl)cc2C1 CC(CNC(=O)CC1CC2(CC2)CO1)CC(=O)NOC(c1ccccc1)C C1(CC)CCN(C(c2cc(C(C)=O)c[nH]2)=O)C1C(=O)N(CCN=[N+]=[N-])CC C1(C(N(CC(=O)NCCC)C)=O)COCCN(C(=O)CC2CC2CC)C1 N(C(=NCCOC)N1CCC2(CC1)C(F)(F)C2(F)F)CC1(CC)CCOCC1 C(=O)(CC1OCc2ncccc21)NC1(C)CC(NC(=O)C(F)=CCCF)C1 C1(CNC(C2CCC(OC)C2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C12CC2 c1(CC(C)N(C(C(=O)N(CC(C)O)CCN(C)C)=O)C)ccc(O)c(F)c1 C1(C(=O)NC(COCC)C(=O)N(CC(F)(F)F)C)COCCN1CC C1(C)(C(C2CCC2)NCC(C)N(C(C(=O)NC(CC)(C)C)C)C)CCCCC1 N1(C(CSCC)=O)CC=C(CCNC(=O)CN(C)C)CC1.c1(S)nnc2ccccn12 c1(C(N2C(CNC(C(CC(C)C)OC)=O)C(C)CC2)=O)cccc([N+](=O)[O-])c1C C1(NC(CN2CC(C)C2)=O)CN(C(c2cccc(NC(N)=O)c2)=O)CC12CCC2 CCCC(C(=O)NC(C)C(=O)OCC)N1CC(O)(Cc2cccnc2)C1 C1(C#N)(CC)CCN(C(=O)C(CC2CC2)NC(C2CCCCCN2C)=O)CC1 Cc1cc(C(N2CCC(CNC(c3cncc(Cl)c3Cl)=O)C2)=O)c2n[nH]cc2c1 C1(NC(c2nn(C)c(O)c2)=O)CC2CC1CN(C(C1CCCCNC1=O)=O)C2 C=CC(C)(CC)C(=O)NCC12CC1CN(C(=O)CC(C)(C)C#N)C2 c1(N2CCC(c3nc(=N)[nH][nH]3)C2)nccc(=NC(=O)N2CC=CCC2)[nH]1 N#Cc1ccc2[nH]cc(CN3CCCN(CS(=O)(=O)CCCCl)CC3)c2c1 c1(C(N(C(CN(C(CC2C(C)=NNC2=O)=O)C)C)C)=O)cc(O)ccc1C N1(C(c2n(C(C)C)ccc2)=O)CCN(C(C23CCCC2CC3)=O)CC(C)C1 N1(C(c2c(-c3c(OC)nccc3)scc2)=O)CCC(NCCCCC(C)C)C(C)C1 c1(C(N(CCN(C(C(COCC)C)=O)CC)CC)=O)cc(C#N)cn1C C1(C)(CNC(c2c(C(=O)OC)[nH]cc2)=O)CCCN(C(=O)C(F)(F)C2CC2)C1 c1(CC)noc(CCC(=O)NCCCCN2CCCC2)n1 C(=O)(CC1=CCN(C(c2cc(F)ccc2O)=O)CC1)N(CC(CC)O)C1CC1 CC(C)C(C)CC(=O)NC(c1ccc(F)cc1)CNC(c1cccc(CO)c1)=O C=CCC(C)(C)C(=O)N1CC2(CC(NC(=O)C=CSNCCc3ccco3)C2)C1 C(C(CC(F)(F)F)NC(c1cc(C)nn1C1CC1)=O)NC(C1N(CC)CCC1)=O N1(C(c2cc(C#N)on2)=O)CCC2(COC(CNC(C3(C(F)(F)F)CC3)=O)C2)C1 C12(C(N3CCC(OC)(CNC(c4csc(Cl)c4)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 c1(NC(C2OCCN(C(c3cn(CC)nn3)=O)C2)=O)cccc(Cl)c1C C(=O)(CCCCCCC(=O)N1CC(NC(c2cn(C)nc2Br)=O)C1)OC N1(C(C2N(C(N)=O)CCC2)=O)CC2(CCCN(C(=O)COCCOCCO)C2)C1 c1(C(=O)NCC2C(NC(=O)CCF)CCC2)cnn2cccc2c1 c1(C(=O)NCCCCC(C)NC(=O)CC(F)(F)Cl)c[nH]c2ccccc2c1=O c1(CCC(=O)NC2CCCN(C(c3cc(C)nnc3)=O)C2)nc2cnccc2[nH]1 c1(C(=O)OC)nc(NC(C2CNCC2c2ccccc2)=O)[nH]c1Br C12(C(N(CC(C)C(C)(C)C)C)=O)CCN(C(C3CCCCC(=O)N3)=O)CCC1C2 C(=O)(C(CC)CCOC)NCc1ncc(C(N(CCCC)CCCC)=O)cn1 c1(CC)oc2ccccc2c1C(N1CC(NC(=O)CC2CCCCO2)C(C)C1)=O c1(C(N(C(CNC(CCN(C(CC)CC)C)=O)C)C)=O)ccc2nc(Cl)nn2c1 c1(C(=O)NCCN(C(=O)CC2CCC(=O)O2)CC)ncnc(CC)c1F C1(NC(C(COC)OC)=O)CCCC2CN(C(C3C=C(C)CS3)=O)CC12 C1(NC(CCCSCCC)=O)CCCN(C(C2CCCN2C(C)C)=O)CCC1 c1(C(=O)NC2CC3C(NC(=O)CCC4CCOC4)C3C2)cc2cccnn2c1 N1(C(C(C)CC(C)(C)C)=O)C2CCCC1CN(C(=O)CCP(C)(C)=O)CC2 c1(CC(C(=O)NC(C#C)CC2CC2)N)cccc(NC)c1 N1(C(c2nn(CC)c(O)c2)=O)CCC2CCCC12C(N1CC(C2CCOCC2)C1)=O C1(N(C(C2CCCN2S(=O)(=O)CC)=O)CC)CCN(C(=O)CP(C)(C)=O)CC1 CC(N=c1ccn(CCS(=O)(=O)N(C)C)[nH]1)c1ncc(C(F)F)[nH]1 N1(C(C(C)=C(CC)C)=O)CC2=C(C1)CN(C(c1c(C)cc(Cl)cc1N)=O)C2 c1(C(N2CC(C)N(C(C3CC3CN(C)C)=O)CCC2)=O)c2c(nn1C)CCOC2 C1(CNC(c2cnc(OCC)c(Cl)c2)=O)CN(C(=O)C(C)=C(C)C)CC(C)(C)C1 Cc1ncccc1C(=O)NC12CC(C1)N(C(c1n[nH]c(C3CC3)n1)=O)C2 C1(CC)C(C(=O)Nc2cnn(C3CC3)c2C)CCN1C(C1CN(C(C)C)C1)=O C1(CNC(C(C)(C)OC)=O)CN(C(c2cc(C)cc(C)c2C)=O)C2(CCC2)C1 N1(C(C2CN(C(N(C)C)=O)C2)=O)CCN(C(C2CCC=CCC2)=O)CC(O)C1 c1(CC(=O)NC2CC(n3cnnc3)C2)cccc(O)c1 c1ccc(C(=O)NC)c(SC)n1.C1(C2CC2)CN(CC2CC2)CCCN1C.CO.OC c1(C(N2CCC(CC#C)(C(=O)NC(C34CC(CO3)C4)C)C2)=O)cc(C)nnc1O C1(CN(C(=O)CNc2nncs2)C)CCN(C(=O)CCN2CCC2)C1 C1(C(=O)NC(C2(CNC(C3(c4ccno4)CC3)=O)CC2)C)CCCN(C)C1 CC1CCC=C1C(=O)NCC(C1CCC1)NC(c1ccc(Cn2ccnc2)o1)=O c1(CN(C(=O)CC2CC3COC2C3)C)ccc(F)cc1 N1(C(C=CCCC)=O)CCC2(NC(c3cc(O)cc(Cl)c3)=O)CC2C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C(O)CC)ccn2cnnc2c1 C1(CNC(C(CCSC)O)=O)N(C(c2cncc(O)c2Cl)=O)CCCC1(C)C Cc1[nH]nc(C(=O)NCC2CC3(CC(NC(C4(C)CCC4)=O)C3)C2)c1[N+](=O)[O-] N1(CCC)CCCC(C(=O)NC2CC(C)(NC(=O)CC3CCOC3)C2)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CC(OC)(CNC(c2nc(C3CC3)ncc2Cl)=O)C1 C1(COC(CCC(C)Cc2ccccc2)=O)CCC2(CCCOC2)O1 C(N=c1cc(C(=O)NOC)nc[nH]1)c1cn(CCCOC)nn1 c1(C(=O)NCCC(C(=O)NCCN2CCOCC2=O)OC)c(C)cccc1O C1(C(NC(COC)=O)CC)CCN(C(=O)Cc2cccc(C(C)(C)C)c2)CC1C CC(C)C(C(=O)n1cc(CN2CCOCC2)nn1)N(C)C.C12C3CN(CC13)C2 N#Cc1ccc(C(=O)NC2CC23CC(NC(c2ccc(NC=O)cn2)=O)C3)s1 c1(N2CCN(c3c(Br)cnc(OC)n3)CC2)cccc2[nH]c(CNC(C)=O)cc12 c1(OC)ncc(C(=O)NCc2ccc(C(=O)NOCCC(C)O)nc2)cn1 C1(NC(c2ncn(C(C)C)c2)=O)(CNC(=O)Cc2cccs2)CCCCC1 c1(C(N(C2CN(C(c3c(OC)cnc(F)c3)=O)C2)C)=O)cc(F)c(F)c(O)c1F c1(C(=O)NCC2N(C(C)=O)CC=CC2)ccc2cc(Br)ccc2n1 c1(C(=O)NC2C3CC(O)C2N(C(C2CCC(F)(F)CC2)=O)C3)cccc2nn[nH]c12 Cc1cc(C(N2CCC2CNC(=O)CCC(C)(C)N2CCOCC2)=O)nc(C)n1 C1(C(N2C(CCC)CCC2)=O)CSCCN1C(=O)CCCC1CCCC1 C(=O)(CCCCC(F)F)NCC1C(CNC(c2nccc(OC)c2)=O)C1 C1(CNC(C2CC(C)C2)=O)CC(C(F)(F)F)CN1C(=O)COCCCF CN=c1[nH]nc(CC(N2CCC(CNC(=O)CN3CCC(OC)C3)CC2)=O)s1 c1(C(N2CCC3CN(C4CC4)C3C2)C(=O)NC(C)C)cc(F)cc(F)c1Br c1(C(N2CCN(C(C(C)OC)=O)C(C)C2)=O)cc2c(Br)cccc2cn1 c1(C(N2CC(NC(C(CC)n3ccnc3)=O)C(OC)C2)=O)ncc(C)cc1F c1(NC(CC2N(c3cc(C)[nH]n3)CCN(C(=O)C(Cl)(Cl)Cl)C2)=O)c(C)cccc1C C(C(F)(F)C(=O)NC(C1CCCC1)CNC(C1CCCSC1)=O)NC(C)=O CC1CC(C#N)(C(=O)NCC2(CNC(C3(O)CC(C)(C)C3)=O)CC23CCC3)C1 c1(C(C(F)(F)F)N(CC(COCC#C)O)C)ccc(Cl)cc1 N1(C(CC(C(=C)C)OCC)=O)CC(NC(=O)C(=O)NC)C2(CCC2)C1 C1(NC(C=Cc2ccc(CC(C)C)o2)=O)CN(C(=O)C(C)CC(F)F)CC1(C)C N1(C(CC(CC)(F)F)=O)CCC(C(=O)NC2CCCCC2CO)=C(F)C1 N1(C(C2C(OCC)C2)=O)CCCC2(C1)CN(C(C1CCc3n[nH]cc3C1)=O)C2 n1(CC)nnc(C(N2CCOC(C(=O)NC(C3CCCCC3)C)C2)=O)c1C C(C(=O)NCCNC(c1cccnc1NC)=O)(C(C)C)OCC C#CCC(C(=O)NCC1(SC)CC1)NC(C1CC(C2CC2)C1)=O N1(C(c2c(C)nc(F)cc2)=O)CCN(C(=O)C(C#N)=CC2CC2)CC(C)(F)C1 C(=O)(C(C)(F)CC1CCCC1)N(CCCNC(C1(O)CC1)=O)C N1(C(c2cnn(C(C)C)c2F)=O)C2CCC1(CNC(C1CC(C(C)C)C1)=O)CC2 c1(C(N2CCC(CCNC(C3=CC(C)(C)C3)=O)C2)=O)cc(O)ccc1[N+](=O)[O-] c1(NC(C2CC(OC)CN2C(C2CCCSC2C)=O)=O)ccc(C)c(F)c1 c1(OC)ccc2nc(C(=O)NC(c3ccccc3)Cc3cccc(Cl)c3)cn2n1 C1(CCNC(CCOC)=O)CN(C(=O)C(c2ccccc2F)F)CCCO1 C12(CNC(CCCSC)=O)CC(NC(=O)CCn3cnccc3=O)(CO1)C2 CN=c1[nH]c(C(=O)NC2CCCC2NC(=O)C(F)n2cccn2)cs1 C(CN=c1[nH]c(=NCc2cncn2CC)c2cccc(F)c2[nH]1)C1(CC)CC1 C1(C(=O)NCCCCn2cc(CCC3CCCCC3)nn2)(OC)CCCOC1 c1(CNC(C2CCCN(C(C(=O)NC3CC3)=O)C2)=O)c(F)ccc(F)c1O C(=O)(C(C(C)(C)O)NC(=O)COC(C)(C)CNC(=O)C(C)CN(C)C)OC c1(C(=O)NCCN(CCOC)C(c2cocn2)=O)ccc(F)c(Cl)c1 c1(C2(C(=O)OCc3cccc(C(=O)OC)c3F)CC2)ccc2ccccc2c1 N1(C(CC(=O)NCC#C)=O)CCC(CC(N2CCCC(C(N)=O)C2)=O)C1(C)C C1(OC)(CSC(C)C(=O)NCCNC(c2ccn(C(C)C)c2C)=O)CCOCC1 c1(C(=O)NCC2N(Cc3nc(C)[nH]n3)CCC2)ccnc(Cl)c1Cl c1(C(=O)NC2C(NC(c3c(CC)cccc3)=O)CC2)ccc([N+](=O)[O-])c(C)n1 Cc1cc(C(N2CC3CC3(NC(C3COCC(C)(C)O3)=O)C2)=O)cc(C)c1C c1(OCC(N2CC(NC(C3C(CC)C3)=O)C(F)C2)=O)cc(C)ccc1Cl C(C(COC)C(=O)NC1CN(C(c2ccc(Cl)cn2)=O)CC1OC)OC c1(C(N2CCC(CCN(C(CCC#C)=O)C)CC2)=O)cccc(C)c1C#N c1(SC)cc(F)ccc1C(=O)NC(C)CCCNC(C1(C)CCCS1)=O N1(C(C2ON=C(C)C2)=O)CCOCC(C(N2CC3CC3C3CC23)=O)C1 Cc1cccc2[nH]c(=NCC(C(C)(C)C)NC(=O)C(c3ccccc3)O)oc12 C1(N(C(=O)CCc2ccsc2)CCC)CCN(C(c2sccc2C2CC2)=O)CC1 CC1(C)C=C(C(=O)NCCCN(C(C23CC(CCO2)C3)=O)C2CC2)C1 c1(C(=O)NC(CCN(C(COCC)=O)C)C(C)(C)C)[nH]nc2c1COC2(C)C C12(CC3(NCc4cc(C(F)(F)F)ccc4)CC3)CC3CC1C2C3O C1(C(N2CCC(C)CC2)=O)CCCN(C(=O)CCP(C)(C)=O)CC1 C1(C(=O)NCC2(O)CN(C(=O)C(Cc3ccsc3)C3CC3)C2)CC(C2CCC2)C1 CN=C1NN(c2cccc(C(N)=O)c2)CC(c2cnn(C)c2)N1C.CC#N N1(C(COC(C)(C)C)=O)CCN(C(C2SCCS2)=O)C(C2CC2)C1 N1(C(C(CCC)OC)=O)CCN(C(C2CCSC2)=O)CC1CC(F)F N1(C(CN(C(COC)=O)C)=O)CC(O)CCC1C(N1CCC(C)C1C)=O CCC(C)(C)C(C)CC(=O)N1CC=CC1CNC(c1nccc2ccsc12)=O C(CN=c1cccc(S(=O)(=O)NC2CC(CO)C2)[nH]1)c1nnc(C)n1C N1(C(C2(c3cccc(F)c3F)CCOC2)=O)CCC(=C(Br)Br)CC1 C1(CNC(CC(C)(C)SC)=O)CC(F)(F)CN1C(=O)C=Cc1nc(C)cs1 N1(C(CN(S(CC)(=O)=O)C)=O)C2CCC1CC(N(C)C(C1CCOC1C)=O)C2 c1(NC(c2c(C3CCCC3)cn(C)n2)=O)ccc(C(=O)N(C)C)cc1C(F)(F)F c1(S)cccc(C(=O)N(CC)CCN(C)C)c1.CCC(C(=O)NC=O)n1ccnc1 C1(NC(COC)CNC(=O)OC(C)(C)C)COCCN1CCCO CC1OC(C)CC1C(=O)N(CCCn1cc(-c2ccnn2C2CCC2)nn1)C1CC1 c1(SCC(=O)NC(CNC(C2(C=C)CCC2)=O)(C)CSC)nc2ccccc2[nH]1 N1(C(C(C)OCC(C)C)=O)CCOCC(CNC(c2cc(C(F)(F)F)on2)=O)C1 c1(C(=O)OC)cc(S(=O)(=O)NC(Cc2cccc(Br)c2)CO)c(Br)o1 c1(CCC(=O)N(CC(=O)O)CC2CCC2)ccncn1 CC1(C)COCCC1C(=O)NCCC(O)CNC(=O)Cn1cncn1 CC1CCC(CNC(c2cccc(N)c2)=O)CN1C(c1ocnc1C1CC1)=O C1(C(=O)NCC(C)=CC(=O)N(C2CCOC2)CCF)CCSC(C)C1 C1(Nc2ncnc(C)n2)CCC2CN(C(=O)CCc3cn[nH]c3)CC12 C12(CC=C)CCN(C1)C(=O)C1CC(C1)CC(=O)N2.C1(C(=O)OC)CCS1(=O)=O N1(C(C(=O)Nc2cncc(SC)c2)=O)CCC(C)C2CCCCC12 c1(CC)sccc1C(=O)NCCOC(C)(C)CNC(C1OCC1(C)C)=O CCC(C(=O)OC)C(=O)NC1CC(CNC(c2ccnn2CC(F)F)=O)C1 c1(NC)ccc(F)cc1NC(C1CSC(C)C1)=O C(C(O)C(=O)NC(C)CNC(c1cc(Cc2ccccc2)[nH]n1)=O)OC C=CC1(C(=O)NCC2(C)CNC(=O)O2)CCN(C(=O)Cc2ccc(O)nc2)C1 N1(C(C(CC)O)=O)CC2(CCN(C(c3c(C)nn(C(C)C)c3C)=O)C2)C1 N1(C(C=CCC)=O)CC(N(C)C(c2cnc(O)n2C)=O)C2(CC2)C1 c1(C(=O)NC2(CNC(=O)CC3CCCCCC3)CC2)cc(Cl)c(Cl)c(Cl)c1O C1(NC(CCNC(CC(C)C)=O)=O)CC12CC(NC(=O)Cc1ccc(Cl)cc1)C2 c1(C(N2CCC(C)(CNC(C3(OC)CC3)=O)C2)=O)ccc(S(N)(=O)=O)o1 N(C1CN(C(=O)CC2CCCCC2C)Cc2ccccc21)C(C=NOC)=O C1(NC(CCNC(=O)NC)=O)CCC2(CC1)CCN(C(=O)Cc1ccc(C)s1)C2 c1(SCC(=O)NC2(C)CCCN(C(c3cnc(Cl)[nH]3)=O)C2)ncnc2[nH]cnc12 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(c2cc(O)cs2)=O)CC(C)C1 N1(C(CCC=C)=O)C2CCC(C2)C1CNC(c1csnc1Br)=O C1(Cn2cc(C3N(Cc4ncc(C)s4)CCC3C)nn2)CCCCC12CCC2 c1(C(N2CC(C(=O)Nc3ccc(C)c(C)n3)C2)=O)cc([N+](=O)[O-])cc(Br)c1F c1(C(=O)NCC2C(NC(c3c(C)snc3)=O)CCC2)ncc(F)cn1 c1(OC)cccc(C=CC(N2CCC(O)(C(C)NC(c3sccc3F)=O)C2)=O)c1 c1(C(C)(C(=O)N2CCC(O)C2)NC(=O)CN2CSCC2=O)ccc(C(F)(F)F)cc1 N1(CC(N2CCC(NC(CSCC#C)=O)CC2C)=O)CCN(CC)C(=O)C1=O C(=O)(C(C)(C)C(C)NC(=O)CCCNC(N)=O)NC(CC=C)C1CC1 N1(N2C(=O)NCC3(COC3)C2)CCCC(S(=O)(=O)N2CCOCC2)C1.C N1(CC(C)C)CCC(C)C1N=c1cc[nH]c(=NCC(F)(F)F)[nH]1 Nc1cccc(F)c1C(=O)NCC1CC1NC(c1ccnc(-c2ccco2)c1)=O CC(=O)CCC(=O)NCCCCC(=O)NCCOCCOC c1(C(C)=O)cn(C)nc1C(=O)Nc1ccc(SCCO)cc1 C(CNC(C1(SC)CCC1)=O)(CCNC(C1C=CCC1)=O)OC C(c1ccncn1)=CC(=O)NC(C1CCN(C(c2c(CC)c[nH]n2)=O)C1)C C=C(C)CN=C(NCC1CCN(C)C1)NCC1(c2cccs2)CCCCC1 N1(C(c2c(Br)cc(OC)s2)C(=O)OC)CCC(C)(O)C(O)C1 C1(NC(CSCC)=O)CCN(C(=O)CN(C(=O)C(C)C)C)CC1F C1(C(C)C)CN(C(c2csc(CO)n2)=O)CCCN1C(c1cnc[nH]1)=O C(c1ccc(=N)[nH]c1)=CC(=O)NCC(CCNC(COCCCCC)=O)O N1(C(C2CCC(C)(CC)O2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)CC(O)C1 C12(OC)CCC(C(=O)NCCCC(C)NC(c3cc(C)c(C)cn3)=O)(CC1)C2 Cc1noc(C)c1C(C)C(=O)NCC1CN(C(=O)C=CC(C)C)CCO1 C1(NC(C(CN(C)Cc2ccccc2)NC(CC(C)C)=O)=O)CCCN(C)CC1 C1(CNC(C(CC)C)=O)CC2(CCN(C(C3(C#N)CC3(C)C)=O)C2)CO1 N1(C(c2cc(C)nc(C)c2)=O)CC2CC(C1)N(C(=O)Cn1cnnc1O)C2 C1(F)(CNC(c2coc(CCN3CCCC3)n2)=O)CN(C(C2(C3CC3)CC2)=O)C1 C1(C(C)C)CN(C(C2CCNC2=O)=O)CC1C(=O)NC1CCC(O)CC1 Cc1ccc(-c2ccsc2)cc1.C(=O)(C1=CCSC1)N1CC(N2C(=O)C2)C1 c1(CNC(=NCC)NCCCCC(C)C)cc(Br)c(OC)cc1F C(=O)(CCC(=O)NCCCN(C1CCSC1)CCCNC(C1CC1Cl)=O)OC n1(CC)ncc(C(=O)NC2CCC(NC(=O)C=Cc3ccc[nH]3)CC2)c1C CCCC(C)(C)C(=O)NC1CC2(C1)CC(NC(c1c(C)nn(CCO)c1C)=O)C2 CC1CCN(C(=O)CCn2cccn2)C(CNC(=O)CC2CC(O)C23CCC3)C1 C1(CC(=O)NCCCOCCCC)CCCCN1C(C1CCC(=O)N1)=O Brc1cccnc1Nc1ccc(N2CCCCC2)nc1 C1(C(N(CCCC)C(C)CC)=O)CCCCC1NC(c1ncccc1O)=O C#Cc1ccc(C(N2CCC(C(N3CC4CCCC34)=O)CC2)=O)cc1 C12CCC(C)N(C1)C(=O)NC2.c1(C(=O)OC)cnc(C)c(N(C)C)c1 CC1CN(C(=O)CN2CCC2)CCC1CNC(c1c[nH]nc1C(F)F)=O c1(C(=O)NC2(C)CCN(C(C3=C(C)CCC3)=O)C2)ccc2cccc(O)c2c1 C(=O)(C(CCC)OC)N1CC(CC(=O)NC2(CC=C)CCCO2)C1 c1(C(N2CC(CNC(=O)Cc3ncccc3F)OCC2)=O)cccc2nscc12 C(=O)(C1CCCc2ncnn21)NCC(C1CC1)NC(=O)CCOCC(F)(F)F c1(C(N2CCC(NC(C)=O)C2)C(=O)NC(CC)C)cc(CC)c(CC)o1 C(=O)(CC(C)C(C)(C)C)N1CC2(C(NC(c3n(C(C)C)cnc3)=O)CC2)C1 C=Cc1cnn(C)c1C(=O)NC(C)CNC(c1cc(CCC)[nH]n1)=O C12(CNC(c3c(C)snn3)=O)CC(NC(C3CCC(C)O3)=O)(CCO1)C2 CS(=O)(=O)c1cc(NC(c2cc(Br)c(Cl)c(Br)c2F)=O)cc(C(F)(F)F)c1 C1(NC(C2CN(S(N)(=O)=O)C2)=O)COC2(C1)CN(C(C1CCC=CO1)=O)C2 c1(CN(C(c2ccc(C)cc2)=O)CC)ccc(F)nc1C.C12CCCC1C(=O)NC2 c1(NC(=O)CC2CCN(C(c3cccc(Br)c3Br)=O)C2)cc(F)ccc1CO N1(C(CC2(OC)CCC2)=O)CC2CC(NC(c3ccc(O)nc3C)=O)CC2C1 C#CC1CCC(NC(=O)C(=O)NC2CCC(CN3CCC(C)CC3)CC2)C1 N(C1CCCn2ccnc21)C(C(Cc1cccc(C)n1)NC(=O)OC(C)(C)C)=O c1(C(=O)NC2C(NC(C3(C)C(C)CCC3)=O)COCC2)coc2ccccc12 C(c1cccc(Cl)c1)=CC(=O)NC(C(C)C)CNC(=O)C(O)Cc1cnc[nH]1 CC(CC(F)(F)F)C(=O)N1CCC(C(C)(C)C(=O)NCC2=CCCOC2)C1 C(c1cscn1)=CC(=O)NC1CCC(CNC(=O)CNC(c2ccoc2)=O)C1 Cc1c(CN(CCNC(=O)OC(C)(C)C)CCO)nnn1C1CCCOC1 C1(CNC(C2N(C)CC(O)C2)=O)CN(C)CCN1C(c1cn(CC(N)=O)nn1)=O c1(OC)ccccc1CC(C)(C)C(=O)NCC1CC1NC(=O)C1=COCC1 C#Cc1ccc(C(=O)NCC2(SC)CC2)c(OC)c1.N12CC(C(F)C1)SCC2=O c1(OC)ccc(NC(=O)N(c2cc(Cl)ccc2N2CCCC2)C(C)C)cc1F N1(C(CC2CC(=O)C2)=O)CCC2CCN(C(c3cc4n(c3)CCCC4)=O)CC12 N1(C(C(CSC)C)=O)CC2CC1CCC2NC(C1CSCC(=O)N1)=O c1(N(c2nc(CO)cs2)C(C)=O)ncc(N(C(=O)CCN2CCCC2=O)C)cn1 c1(C(=O)NCC(=O)OC(c2ccccc2)CCC)ncn(C)c1C CCC(C)C(O)C(C)C(=O)N(CC(C)NC(=O)CC(C)c1cnn(C)c1)C C#CCC(CC(=O)NC(C1CCCC1)CO)NC(=O)COCCCC C1(NC(C2(CC#C)CC2)=O)CN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC2CC12 CC(C)CCC(=O)NC(C(C)NC(=O)CCOC1CCOCC1)C(C)C N1(C(Cn2ccc(C)n2)=O)CC2CCC1CN2C(c1ccc(=O)n(CCF)n1)=O C1(NC(CC2N(CC)CCC2)=O)CN(C(c2ncoc2C2CCC2)=O)CC1F CN=c1[nH]cc(C(=O)NCC2CCC2NC(C2C3COCC23)=O)s1 O=C1Cc2cc(C(=O)NC3CCN(C(=O)C(=Cc4c[nH]cn4)F)CC3)ccc2N1 C1(C(=O)NC(C)CC2CCCC2)CCN(CC(=O)NCCCOCCO)CC1O N1(C(c2n(C)cc(C(=O)O)n2)=O)CCC(C2CCCC23OCCO3)C1 C1(CC)CN(C)C(=O)CN1C(=O)C(c1ccccc1)NC(c1cc[nH]c1)=O N1(C(CCCOCC)C(=O)NC)CCC(C)(C(=O)Nc2conc2C)C(F)C1 N1(c2nc(N3CC(C#N)OCC3)c3c(n2)[nH]cc3)CCOC2(CCSC2)CC1 c1(C(=O)NC2C3CN(Cc4c(C)nn(C)c4Cl)CC32)cc(F)c(F)c(F)c1F c1(C(=O)NC2CC(CNC(CCc3onc(CC)n3)=O)C2)cc(C)c(Br)o1 N1(C(c2cc(C(C)C)on2)=O)CCC2(CC(NC(=O)C(F)=C3CCCC3)CO2)C1 C(=O)(CCCCNC(C1(CC)CCCO1)=O)NCC=C=C S(=O)(=O)(c1ccc(Cl)s1)N1CCC(CCN2CC(C)(c3nn[nH]n3)C2)CC1 C1(NC(C2=C(C)CCCC2)=O)CCCCC12CCCN(C(c1cc(O)cs1)=O)C2 c1(C(=O)NCCN(C(c2cnc(=NC)[nH]c2)=O)C)cc(C)cc(OC)c1C c1(C(=O)NC2CCN(C(C3CCOCC3)=O)CC2)csc(=NC2CC2)[nH]1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCOCC(C)(CNC(=O)C2=NNC(=O)CC2)C1 C1(CNC(C(CC=C)CC)=O)CC2CCC(C1)N2C(C1CN2CCCN1CC2)=O Cc1c(C(N2CC(NC(=O)C(C)CF)CC2C)=O)cnn1-c1cccc(Cl)c1 CC1=C(C(=O)NCc2ccc(CNC(C3CCCC3CN(C)C)=O)cc2)CCC1 c1(N(C(C)C)C)cc(Br)ccc1S(=O)(=O)NCC(C)C1(CO)CC1 N1(C(c2cccc(C3CC3)c2)=O)CCCN(C(=O)C(c2ccccc2F)F)CC1 C1(=C(F)CNCC=CC(=O)OCCc2cn(C)nc2C(F)F)CC1C1(C)COC1 C(=O)(C(C)(C)C(C)C)NCC(C1CCC1)NC(C(C)Oc1cccc(CO)c1)=O c1(C(=O)NC2CCCCC2CNC(C23CCC(CO2)C3)=O)cc(O)nc(O)n1 C1(CCC)CCCN1C(C1C(NC(=O)COCCCOC)C1)=O Cc1cc[nH]c1C(=O)NC(c1cccnc1)C(=O)NCC1(C(N)=O)CC1 C(=O)(C(C)(F)C(=O)N1CCN(C(=O)C(C)Oc2ccccc2)CC1)OC N1(C(c2ccc(O)c(Br)c2)=O)CC2(CCC(NCc3ccc(I)o3)C2)C1 c1(NC(=O)NCC2N(Cc3ccccc3)CC2(C)C)ncn2c1CCCC2 C(C(C)C)(C(C)(C)O)NC(CC1(OC)CN(C(C2(C(C)=O)CC2)=O)C1)=O C1(C(=O)NC(CNC(C(C(C)C)NC(C)=O)=O)(C)CO)CN2CCCN1CC2 N1(C(CC2C(C)(C)CCO2)=O)CC2(COC(CNC(c3ccc(CO)o3)=O)C2)C1 c1(C(=O)NC2(C)CC(NC(C3(C4CC4)CC3)=O)C2)cc2cc(Br)ccc2cn1 c1(C(=O)NC2(CCNC(C3CCCCS3(=O)=O)=O)CC2)ccc2c(c1)CNC2=O N1(C(c2ccc(C)c(CO)c2)=O)CCC(C2CN(C(C3CNC(=O)C3)=O)C2)C1 C(CCN=[N+]=[N-])NC(CN(CC)CC1(C(=O)N(C2CCC2)C)CC1)=O C#CC1CCCC(C(N2CC(CC(=O)Nc3ncccc3Cl)C(C)C2)=O)C1 C1(C(N(C)C(C2CC2)C2CC2)=O)CN(C(C2(F)CCCC2)=O)CC1(C)C C1(C(=O)NCc2c(C(=O)NC(C)CC3CC3)cccn2)CC2CCC(C1)C2 CC1CCCC1CC(N1CC(O)(CN(C)C(C2CC2(C)C(F)F)=O)C1)=O Cc1coc(C)c1C=CC(=O)NCC1(F)CCCN(C(=O)C(C)NC=O)C1 N1(C(c2ccc(C)cn2)=O)CC2CCCC2C1C(N1CC2C(C1)C2(C)C)=O C(=O)(C1CCOc2c(F)cccc21)N(CCCNC(c1cc(F)n(C)n1)=O)CC c1(OC)ccc(C(=O)N(C2CN(C(=O)C(F)CC3CCC3)CC2F)C)cn1 c1(C(=O)NC2CC(NC(=O)CCCC3CC3)CC2O)cnc2[nH]nc(O)c2c1 c1(C(=O)NCCCC(C)NC(c2cccn2C)=O)noc2ncccc12 c1(SC)ccc(OC(C)C(=O)NC2CCC2NC(=O)Cc2ncoc2C)cc1 C(=O)(C(C)CC(F)(F)F)NC1CC2(CC(NC(c3cc(OC)cc(=O)o3)=O)C2)C1 C1(C(=O)NCCC(=O)OCC)CN(C(C2CC(C)(C)C2)=O)CC1OC C1(NC(C(=O)NCC2CC2Br)=O)CC(N=c2[nH]nc(CC3CC3)s2)C1 N1(C(C(=O)NC(C)C)C)Cc2cc(Br)ccc2CC1C C1(COC)CN(c2nc(N(CC(C)(C)C)C)nc3c2SCC3)CCC12CCCC2 C(=O)(C(F)C(=O)NC(Cc1cnc[nH]1)C(=O)NCCCCCC1CC1)OCC c1(C(=O)NCC(F)(F)F)ccc(F)c(Cl)c1F.C1(OC)CC2N(C1)C2.C1(=O)CO1 c1(OC)c(C(=O)NC2CC(NC(c3cncnc3C)=O)C2)cccc1Br N1(C(C(C#C)(C)C)=O)CC(NC(=O)C(CCC)OC)C2(CCOCC2)C1 c1(OC)ccc(S(=O)(=O)NC2CC2C(=O)Nc2cc(Cl)nc(Cl)c2)cn1 c1(C(=O)NCC(C2CCC2)NC(C(C=CC)O)=O)ccc(C2CCC2)nc1 Cc1cccc(C(N2CCC(NC(=O)CC3CN(C)C3)CC2C2CC2)=O)c1N CCC(C)CCCCC(=O)NC(C)CCC(=O)N(CCO)CC c1(OC)ccc(Cl)c(C(=O)NCC2CC2NC(c2cnn(C)c2C(C)C)=O)n1 C1(C(N(C2CCCN(C(=O)Cn3cc(C#N)cn3)C2)C)=O)CC2(C1)CC(O)C2 c1(C(=O)NC2CCN(C(Cc3nnc(C)o3)=O)C(C)C2)cc2c(C)n[nH]c2[nH]1 C1(C(=O)NC(C#C)CC)C(O)CCN1C(=O)C(O)CN1CCCC1 c1(C(N2CC3CC(NC(c4[nH]cc(C)c4)=O)C3C2)=O)cc2c(nc1O)CCSC2 C(CC(C)C(=O)NCC(c1ccccc1)NC(=O)Cn1ncccc1=O)=CC C1(NC(CNC=O)=O)CC(O)CN(C(c2cc(NCC3CC3)ncc2Cl)=O)C1 Cc1cccc(C(=O)NCC2N(C(=O)C3=C(Cl)CCC3)CCC2(C)C)c1F N1(C(C)C)C(=O)COCC1C(=O)NCCOCCNC(=O)C(c1ccc(Cl)s1)C C1(CNC(C2N(CCC)C(=O)CC2)=O)CCN(C(=O)COCCC(C)C)C1(C)C N1(C(CN2C(C)CCC2)=O)CCC(C(=O)NC2CCCN(O)C2=O)C(C)(C)C1 CC1CCC(CNCC2(N)CC(O)C2)C1 N1(C(c2c(COC)cco2)=O)Cc2n[nH]cc2C1C(=O)NCC1(C2CC2)CC1 N1(C(CCOC(C)=O)=O)CCN(C)C(CNC(c2cc(Br)n[nH]2)=O)C1 N1(C(C2C(C3C(C)C3)C2)=O)CCC(C2CCCN(C(=O)C=Cc3ccco3)C2)C1 Cc1ccc(CCC(N2CCN(C(c3cc(Cl)cnn3)=O)C3CC23)=O)c(C)c1 C1(OC)(CNC(c2ccnc(CO)c2)=O)CCN(C(C2(C)CCC(=O)N2)=O)C1 C1(C(N(CCCC(=O)NCC(C)Cn2cccn2)C)=O)CCS(=O)CC1 c1(NC(=O)NC(CC)C(=O)NC(c2cccnc2)C(C)C)ccccc1C N1(C(C=C(C)C(C)(C)C)=O)CC(CNC(=O)C(C)OCC2CC2)C(O)C1 c1(C(=O)NCC2C(C)CCN(C(C3C=CC=CC=C3)=O)C2)ccc(N)c(Cl)c1O c1(C(N(CC(C)NC(COCC)=O)C)=O)n[nH]c2cc(C)ccc12 c1(C(N2CCC(OCCNC(C=COCC)=O)C2)=O)ccc2ccc(C)cc2n1 c1(C(=O)NC2CC(NC(C3(CC#C)CCOCC3)=O)C2)ccc2c(c1)CCC2 C(C)(C)(CCC(=O)NC1CCC2CC1CO2)NC(COCC(C)C)=O c1(C(=O)NC2CC3CC2CN3)ccc(-c2ccncc2)nc1O N1(C(c2ccc(C#N)cn2)=O)CCCC2(CCC2NC(C2CC(F)C(=O)N2)=O)C1 C(c1ccc(F)c(Cl)c1)=CC(=O)NC1C(NC(c2c(C)ccc(Cl)c2)=O)CC1 CCCCCC(CCCCC)CC(=O)NCCCNC(=O)COc1cnn(C)c1 N1(C(CS(C)(=O)=O)=O)CCC(CO)C(NC(=O)C(O)Cc2ccccc2Cl)C1 C1(C)(CNC(CCCNC(C)=O)=O)CCN(C(C2OCCC2(C)C)=O)C1 Cc1cc([N+](=O)[O-])c(C)cc1C(=O)Nc1ncc(NC(=O)C2=NNC(=O)CC2)s1 C#Cc1ccc(C(=O)NC23CC2CN(C(c2ncnc(C)c2C)=O)C3)c(F)c1Cl C=CCC(C)(C)C(=O)N1CC(OCCOC2(F)CCN(C(=O)CC)C2)C1 C1(NC(C(C)(C)C2CCOC2)=O)CC2(C1)CC(C(N1CCC13CCCC3)=O)C2 CC(C)(CNC(C1CC2(C1)CC21CC1)=O)CC(=O)NCCCN1CCCC1=O c1(C(C(=O)NCC(CNC(=O)CCc2nc[nH]n2)F)NC(N)=O)ccccc1 c1(OC)ccc(C(=O)NCCN2CCN(C(c3cccs3)=O)CC2)c(C)c1 N1(C(Cc2nc(C)oc2)=O)CCC2CC12C(=O)NCc1cn(C)cn1 c1(C(=O)NCC2CC3(CCC3)CN2C(=O)CC=C(Cl)Cl)cc2cccn2cn1 c1(C(=O)NC2CCN(C(c3c(C)[nH]nc3Cl)=O)CC2O)coc(S(N)(=O)=O)c1 C(=O)(C(C)(C)CSc1ccccc1)NCC1C(NC(CCSCC#C)=O)C1 c1(CS(N)(=O)=O)cccc(=NC(=O)CC2CC3(CCOCC3)CO2)[nH]1 c1(C(N2C(C)(CNC(CSc3c(C)cccc3)=O)CCC2)=O)ccc(Cl)c(O)c1 CCC(C)C(=O)C(=O)N1CCCC(C(=O)NCC(CC)C(C)C)(CC)C1 c1(CC)cnc(C(N2CC(NC(=O)C=C3CCC3)C3CC23)=O)cn1 C1(NC(CCSCCCC)=O)CN(C(=O)CCCC2CCCC2)C(C)(C)C1 C1(C(=O)NCC2CCC(C)C2)(NC(Cc2cn(CC)nc2)=O)CCN(C)C1 N1(C(CSCC#C)=O)CCC2(CCC(NC(=O)C3=CCCC3)C2)CC1 C1(C(=O)NC2CCC(CCNC(=O)CSC(F)F)C2)CCCCCCC1 c1(NCCCC(N2CCN(c3ccccc3F)CC2)=O)ccc2cncn2c1 N1(C(CSCCC)=O)CCC2(CC(C(N3CCCC3C(=O)OCC)=O)C2)C1 C#Cc1ccc(Cl)c(C(=O)N(CCCNC(c2csnc2OC)=O)C2CC2)c1 C12(CNC(c3c[nH]c(C)c3C)=O)CCC(CC1)N(C(=O)CSC(C)(C)C)C2 N1(C(CCC(=C)C)=O)CC(NC(=O)CC2=CCCC2)CCC1C CC(=O)CCCC(=O)N1CCC(C(=O)N(CC(O)C2CCC2)C)C1 N1(C(C(C)(C)CC(F)F)=O)CC2(CCCCN(C(=O)CCc3ncc[nH]3)C2)C1 C1(NC(c2cnc(CC)[nH]2)=O)CC(O)CN(C(=O)CCc2cncc(C)c2)C1 COn1cnc(C)c1C(=O)NCCC1(O)CCN(C(=O)C(c2csc(C)n2)=O)C1 C1(C(=O)NC(C2(O)CCN(C(C=C(C)C(C)C)=O)C2)C)CC2(C1)NC(=O)NC2=O c1(C(N(CCCCCNC(C2CCCC(OC)C2)=O)C)=O)nccc2n[nH]cc12 N1(C(C2(C3CC3)CN(C(CC(C)C(F)F)=O)C2)=O)CCOCC(C)(O)C1 C1(CC)CN(C(C2CCC(C#N)CC2)=O)CCN1C(c1ccc(C(N)=O)cc1)=O c1(OC)cc(OC(F)F)c(F)cc1[N+](=O)[O-].C1(C(F)(F)F)CC(=O)N1 CC1CC(NC(c2cn[nH]c2)=O)CCN1C(c1csc(-c2ccncc2)n1)=O c1(OC)cccc(CS(=O)(=O)NC2CC2C(N2CC(CS(C)=O)C2)=O)c1 CCC(CC)(CC)C(=O)N1CC2CC(NC(C3(N(C)C)CCC3)=O)CC1C2 C1(CNC(Cc2c(C)nc(SC(F)F)s2)=O)CCN(C(c2csc(O)n2)=O)C12CC2 C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CC(NC(C2CCCC(O)C2)=O)CC1O C1(COC)CN(C(c2cnc(Cl)c(C)c2)=O)CCN1C(C1CCSCC1)=O c1(-c2ncnn2C(C)COC)nc2ccccc2[nH]1.c1(OC)cccc(OC)c1Cl c1(C(N(C)CC2(NC(c3cc(C4CC4)ns3)=O)CC2)=O)ccc(Cl)cc1 c1(OC)cc(C(=O)NCCOCCN(C(=O)C(C)C2CCCO2)C2CC2)ccc1Cl c1(C(N2CCC(C)(C(=O)NCC#N)CC2)=O)c[nH]c2cccc(F)c12 c1(C(N2CC(O)CC2C)C(=O)NCC)cccc2c1COC2=O FCCCN=C(NCc1nc(CSC)cs1)N1CCC(C(F)(F)C(F)(F)F)C1 S(=O)(=O)(c1ccc2c(c1)CCO2)NC1C(OC)CN(C(c2cnco2)=O)C1 C(=O)(CCCCN(C(=O)Cc1ccn(C)c1)C)NC(c1ccnn1C)CC C(=O)(C(O)CC(C)(C)C)NC1CC2C(NC(c3c(C)cco3)=O)C2C1 c1(CC)nc(=NCC(C2CC2)NC(=O)CC2(c3ccccc3)CC2)s[nH]1 N1(C(c2c(C)nns2)=O)CC2CCC1C(NC(c1cnc(S)n1C)=O)C2 N1(C(CC2C(C)C2)=O)CCSCC1CCNC(C1(CF)CC1)=O C=C(C)CCC(=O)NC1C=CCN(C(c2cc(C(F)F)ncn2)=O)C1 C1(C(=O)NC2CC(CNC(COCc3cc(C)on3)=O)C2)CN(C)CCN(C)C1 CC(C)(CC#N)C(=O)N1CCN(C(c2ccc[n+]([O-])c2)=O)C(CN(C)C)C1 N1(C(C2(c3ccccc3Br)CC2)=O)CC(C(N2CC3CCC(C2)O3)=O)CC(F)C1 N1(C(C(C)O)=O)CCOC2(CCCN(C(c3cc(Br)cc4nn[nH]c34)=O)C2)C1 c1(C(=O)Nc2ccc(C)cc2C(N)=O)coc2c1CN(C(=O)C1CC1)C2 Cc1ccc(Cn2cc(C(C)(C)NC(C3CCCO3)=O)nn2)cc1 c1(OCC=C)ccc(CC(=O)NC2CC2CNC(c2cncn2C)=O)cc1OC c1(CC(=O)NCC(C(C)C)NC(CC(C)OC)=O)cnc2c(C)cccn12 C1(C(N2CC(OCC(=O)NC3(COC)CCCCC3)C2)=O)CC(=O)NC1(C)C n1(CCC(=O)OCC(=O)NC23CC4CC(CC(C4)O2)C3)ccc2cc(Cl)ccc12 N1(C(C=Cc2ccc(OC)cc2F)=O)CCNc2ncc(C)cc21 C=CCCC(C(=O)N1CCCCC1CC(N)=O)NC(C1OC2CCC1C2)=O c1(-c2ccc(NC(C3(C)CCN(CCOCCO)C3)=O)o2)cn2ccccc2n1 c1(N(C)C)cc(C(=O)N(CCNC(C2(O)CC(C)(C)C2)=O)CC2CC2)cc(Cl)n1 Cc1cccc(CCC(=O)NC(C)CCCCNC(=O)CC2CC(C)(C)CO2)c1 c1(C(=O)NCC2N(C(c3[nH]c(=NCC=C)sc3)=O)CC2)cc2c(cn1)CCCC2 C(=O)(C#Cc1ccccc1)NCCN(CCC)CC c1(C2(C(=O)NCCCNC(C(C)OCCC#C)=O)CC2)ccc(Br)o1 C#Cc1cccc(C(N2CC3CC3(CNC(C3(N=[N+]=[N-])CC3)=O)C2)=O)c1Cl C1(F)(CNC(C(C)NC(N)=O)=O)CCN(C(=O)Cc2cccc(Cl)c2Cl)CC1 c1(-c2cnc(N3CCN(Cc4ccn(CC)n4)CC3)nc2)ccc(C#N)c(Cl)c1 Cc1nnc(O)c(C(N2CC(CNC(c3ccnn3CC#N)=O)C2)=O)c1C c1(C(N(CCC(C(C)C)NC(C2CCN(C)C2)=O)C)=O)ccn2c1CSCC2 C1(OC)CC2(C1)CC2NC(=O)C(CCF)NC(=O)C(=O)N(C)C C(C(=O)NCC1CC1N(C(=O)C=CC(C)=O)C1CC1)N(C)CCO CN1Cc2ccccc2C1CNC(=O)NCc1ncc(C2CCCCO2)s1 C1(NC(C2C(C)OCC2)=O)CN(C(C2CC3(CCC3)CO2)=O)C2CCCC12 N1(C(CCC)=O)CCCC2(NC(c3cn(C(C)C)cn3)=O)CCCC12 CC(CC(N)=O)C(=O)NC(c1ccccc1F)CNC(=O)CN=S(C)(C)=O C1(C(N2C(C)CC(CC(=O)NC3C(CC)(CC)C3)C2)=O)CN(C)C(=O)C12CC2 c1(C(=O)N(CCOCCCC)C2CC2)ccc(-c2ccccc2)cn1 n1(CC(=O)NC(C2(C(=O)NC(C(=O)NC)C)CC2)C)cc(Cl)cn1 c1(OC)ccc(N(C)C(=O)N(C)C)cc1Cl.c12ccc(cc1)OC(=O)C2 C1(NC(c2cnc(OC)nc2)=O)CN(Cc2cccc(F)c2O)CCC1C S(=O)(=O)(c1ccc(CBr)cc1)NC1CN(C(C(C)(C)CO)=O)CC12COC2 C(CCC(C)C)(C(=O)N1CCCCC1CO)NC(C(COC)N(C)C)=O CC1=C(C(=O)N2CC3CC2C3NC(c2cc3c(nn2)CCC3)=O)CCC(C)(C)C1 N1(C(C2(SCC)CC2)=O)CCC2(CC(NC(c3cc(Br)n(C)n3)=O)C2)C1 CCCN(OC)C(=O)C1C(NC(=O)Cc2cccs2)C1(C)C N1(C(CC(C)c2ccco2)=O)CC2(CCCC(CNC(=O)CO)O2)C1 c1(C(C)C)cccc(N=c2scc(-c3ccoc3)n2C(C2CC2)C2CC2)c1 Cc1nc2n(n1)CCN(C(c1oc(NC(=O)COC3CCCOC3)nc1C)=O)C2 c1(C(NOCCCOC)=O)ccnc(CNC(c2cc[nH]n2)=O)c1 N1(C(c2nc(C(C)C)no2)C(=O)NCCCC)CCN(C(C2CCCO2)=O)CC1 C1(C(=O)NCC(C)C#N)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 c1(OC)cc(-c2ccc(F)c(CN(CC(C)(C)O)C)c2)ccc1C N1(CC(=O)NCC2(NC(C3CC(CC)OCC3)=O)CC2)OC(C)(C)CC1=O c1(OC)ccc2c(c1)S(=O)(=O)N(C(C)C(c1c[nH]cc(C(F)(F)F)c1=O)=O)C2=O C(CN=C(NCCC(C(F)F)SC)NC1CCCOC1)N1CCCS1(=O)=O.C=CCO C1(NC(C)CCN(C(=O)CCOCC(F)(F)F)C)CCOC1C(F)(F)F C#Cc1cc(F)c(C(N2CC(NC(C3(COCC)CC3)=O)CC(C)C2)=O)cc1F c1(NC(C(=O)NC(CCC)CCc2ccccc2)=O)ccc(Cl)c(C(F)(F)F)c1 N1(CCOCCOCC)CCN(C(=O)CSC2CCC2)CC(O)C1 N1(C(c2c(C)ccnc2Cl)=O)CC=C(CCNC(c2cccnc2C)=O)CC1 C1(C(C)NC(=O)CSCC(N)=O)CCN(C(=O)CCCNS(C)(=O)=O)C1 c1(-c2cn(CCCC(=O)N(C3CCCC3(F)F)CCO)nn2)ccc2ocnc2c1 C(c1ccccc1)=C(CC)C(=O)NC1(C)CN(C(=O)Cc2nncn2C)C1 CCCCC(CNC(C12CC1COC21CC1)=O)NC(C12COC(COC)(C1)C2)=O C1(CC(=O)N(C)CC2(OCC)CCC2)C2CCC(C2)N1C(=O)C(O)SC C1(NC(C(CCC2CC2)NC(=O)Cc2cnco2)=O)CC2CCC(C1)S2 C1(NC(C2C(C)CC2)=O)CC2(C1)CC(C(N1C3CSCC1C3)=O)C2 C(=O)(C(F)CC(C)(C)NC(=O)CN(C)CCOC)NC(c1ccccn1)CC N1(C(c2cc(CCC)on2)=O)CC2(C(N3CC(O)CCC3C)=O)CCC1CC2 C1(N(C(C)C(=O)N(CC(C)CNC(C23CC(C)C2C3)=O)C)C)CCCCCC1 N1(C(CC2CCC(=O)NC2)=O)CC2CCC(NC(=O)C3=C(Cl)CCCC3)(C2)C1 C(CCC(C)(C)C(=O)NCc1nn(C)c(=O)n1C)NC(C1C(C)(CC)C1)=O Cc1sc(CNC(C)CN2C(=O)CNC2=O)c(Br)c1C N1(C(Cc2c(C)non2)=O)CC(C(=O)NCc2cccnc2Cl)CC(C)(C)C1 C=CCC(CCCCC)C(=O)NC1CCN(C(=O)CNC(=O)C(C)C)CC1CC c1(C(=O)NC(C(N2CCN(CC(C)O)CC2)=O)(C)C)cc2ncccc2[nH]1 Cn1cc2ccc(NC(C3CC3NCc3cc4cccn4cn3)=O)cc2n1 c1(CC)[nH]nc(Cl)c1C(=O)NCCC1CCC(NC(=O)CCCSC)C1 c1(CC(C)NCC(=O)Nc2cc(Br)ccc2N)ccccc1[N+](=O)[O-] Cc1sc(C(=O)NC2CCCCC2NC(c2cncnc2)=O)nc1Br Cc1nc(C(N2CCCCC2CCCNC(C2(C)CC(C#N)C2)=O)=O)cn1C N1(c2cc(NCc3nccc4ccsc34)ncn2)CC2CCCC2C12CC2 C1(NC(CC2(C)CCN(C(c3c(C)oc(CO)c3)=O)C2)=O)CN2CCC1(C)CC2 n1(CCNC(N(C)CC)=O)nc2ccccn2c1=O.C1(C=O)(CO)CCC(C)CC1 N1(C(CCc2ccn(C)n2)=O)CC2CC1CC2CNC(C1CS(=O)(=O)C1)=O C(=O)(C(C#N)C(C)(C)C)N1CC(O)(CNC(c2cc(C(=O)OCC)c(C)[nH]2)=O)C1 C1(NC(c2ccnc(F)c2)=O)CCCN(C(=O)CCCc2cccc(Cl)c2)C1 CC1(CNC(=O)CN2CCCNC2=O)CCC(NC(C2CC(n3cnnc3)C2)=O)C1 C1(C(=O)NCC23COC(CO)(C2)C3)CCC2CCCCC2C1 c1(OCC(=O)NCCCCCN(C)C(C2CC2C#N)=O)cccc2cccnc12 C#Cc1cccc(C(N2CCN(C(=O)C(Cl)=CCl)CC2C2CCC2)=O)c1 c1(C(N2CC(C(=O)NC)OCC2)C(=O)NCCC#N)cc(I)ccc1OC CC1OC(C)(C)OC1(C)C(=O)N(CCCNC(c1cn(C)nc1C(F)F)=O)CCO C(=O)(C(C)(O)CC(F)F)NCC1(C(F)(F)F)CC(C)(C)C1 N1(C(C=CC2(C)CCOCC2)=O)CCC2CCC(NC(=O)CC3CC(F)C3)C1C2 N1(C(C)=O)CC(O)CC1C(N1CCC(N(C(=O)C=C2CCC2)CCO)C1C)=O N1(C(c2ccc(CSC)o2)C(=O)NCCOC)CCCC(O)(C(F)(F)F)C1 C(=O)(C(CC(C)C)NC(N)=O)NCCC1CC(CNC(CC2(OC)CC2)=O)C1 c1(C(=O)NC2CN(C(c3scc(C)c3C)=O)C(C)C2)cc[nH]c(=N)c1[N+](=O)[O-] C1(NC(C2C(C)(C)CCCC2)=O)CC1C1CCCN(C(C23CCCCC2C3)=O)C1 Cc1ccc(OCC(=O)NCC2(F)CN(C(C3CC4CCC3CC4)=O)C2)cc1C C1(NC(C(C)(O)C2CCC2)=O)COC2C(NC(c3cccc(=O)o3)=O)COC12 C(=O)(C(C)(C)CS(=O)(=O)N=S(C)(=O)c1ccccc1Cl)Nc1c(OC)cc(Cl)cc1 n1(CCC(=O)OCC(=O)NCc2c(C)ccs2)ccc2cc(Cl)ccc12 C1(C(=O)Nc2scc(NC(=O)Nc3ccccn3)n2)CC2(C1)C(CO)C21CCC1 N1(C(C(c2ccco2)NC(C(C(C)C)SCC)=O)=O)CCCC2COCC12 c1(C(=O)NCCC(C)NC(Cn2ccc(C)cc2=O)=O)cc2cc(F)ccc2[nH]1 C(=O)(CC(F)(F)C(F)F)N(C1CCN(C(C)=O)CC1)CC=C c1(OC)cc(C(N2CCC(CCNC(=O)COC)C2)=O)cnc1OC1CCC1 C1(C(N2CC(OC)C2)=O)C=CCN1C(=O)CC1CC(C)C1 c1(N(CCC)Cc2cccnc2)nccc2c(C)cccc12 N1(C(C2CN(C(=O)NC)C2)=O)CCC2(CC2NC(c2cc(Cl)c(Cl)s2)=O)C1 C(=O)(CC1=CCCCC1)NCC1C(NC(c2c(C)c(C(C)C)on2)=O)CC1 N1(C(CC(C)(F)F)=O)CCOC2(CCC(NC(=O)CC(C)(O)C(F)(F)F)CC2)C1 c1(C(=O)NCC(C)N(C(c2ccc(OCOC)cc2)=O)C)cccc(N)c1F N1(C(CCC(=C)C)=O)CC2(CCCC(CNC(=O)CCC3CCN(C)CC3)O2)C1 CC1(C)CCN(C(c2sc([N+](=O)[O-])cc2Cl)=O)CC1NC(C1CC1CF)=O C1(CC)CCCC1(c1nnnn1C)NCCCc1ccnc(C)c1 c1(C(=O)NC2CC2CNC(=O)C(F)n2ccnc2)ccc2oc(O)nc2c1 C(C)(CCN=c1ccnc[nH]1)NC(c1c(C)cc(F)nc1)=O C1(NC(CCC=CC)=O)CCCC12CCN(C(c1ccc(N)c(SC)c1)=O)C2 C1(CNC(c2cc(CC)[nH]n2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1(F)F C1(N(C(C(C)=C2CC2)=O)C)CCCN(C(=O)C(C)Sc2cccc(C)c2)C1 Cc1cccc(-c2ncc(NC(=O)CN3CCC(C(C)(F)F)C3)s2)c1 c1(NC(c2ccc(-c3ccc(COC)cn3)cc2)=O)cc(Cl)cc(Cl)c1F N1(C(c2ccc(C(F)F)s2)C(=O)NCCOC)CCN(CC(F)F)CC1 C1(CC=C)(NC(C2CC(C)(C)CO2)=O)CCCN(C(c2nc(=N)cc[nH]2)=O)C1 N1(C(CCSCCC)=O)CCN(C(c2c[nH]ccc2=O)=O)CC(CO)C1 N1(C(C(=O)NC2COC2)CCC2CC2)CCC(O)C(O)C1 Cc1cc(C=O)[nH]c1C(=O)NCc1cc(-c2ccccc2)no1 CCCC(C(=O)N=c1cc(C)o[nH]1)NCC(O)COc1cc(C)cc(C)c1 C1(CNC(CCN(C(CCC)C)C)=O)COCC1NC(c1nnsc1C)=O N1(C(C2C(=C)C2)=O)CCCC1(C(=O)N(CC(CC)(CC)OC)C)CC CC(CC(=O)NCC1CC2CN(C(C34CCC(C)(CC3)CC4)=O)CC12)C(C)(C)C c1(C(=O)NC(C2(O)CCN(C(C3C(CC)C3)=O)C2)C)cnc2c(cnn2C)c1 N1(C(c2ccn(CCCC)n2)=O)CC2CCCC2(NC(C2CCS2(=O)=O)=O)C1 c1(C(=O)NCC2CCN(C(C3C(C)OCC3)=O)C2)sc(=N)[nH]c1C1CC1 N1(C(C2C(CCC)CN(C(C3CCCO3)=O)C2)=O)CC2(CCCCCC2)C1 C1(C)(CC)CN(C(C2CC23CC(NC(C2C(C)C2C)=O)C3)=O)CCO1 C1(NC(C2CCC(C)C2)=O)CCN(C(=O)C(C)N(C)C(C)=O)C12CC2 C(=O)(CCCC(F)F)N1CC(C(C)NC(=O)CSc2cnn(C)c2)OCC1 C1(C(=O)NCC(C)(C)O)CC2(CCN1C(C1CC(=O)CC(=O)N1)=O)CC2 c1(C(=O)NC2C(C)(C)CN(C(c3cnc[nH]c3=N)=O)C2)ncn2c1COCC2 CCC(C)(C)C(O)C(=O)NCCC1CCCCN1C(c1ccn(CC(F)F)n1)=O C=Cn1nncc1C(=O)N(CCN(C)C(c1ncn(CC)n1)=O)C(C)C CN1CCC(CC(=O)NC(CNC(=O)COc2ccc(F)nc2)CO)CC1 n1(CC)cnc2nc(=NC3CCC4(CCCCC4)C3)[nH]cc12.C(N)=O c1(C(N(C(C)C(N2CCSCC2CO)=O)CC)=O)cccc(C)c1 c1(OC)ccc2[nH]c(C(N3CCOCC3CNC(=O)CC3CSC3)=O)cc2c1 c1(OC)c(C(=O)NC23CC2CN(C(C2CCOC2)=O)C3)cnc2ccccc12 CC1OC2(C)CC1(C(=O)NCC1CC(NC(C3CCS(=O)(=O)CC3)=O)C1)C2 CC1C=C(C(=O)NCC2CCCN2C(=O)CCCn2ccccc2=O)CC1 c1(C(=O)NCC2(NC(CC3CCCN(C)C3)=O)CCOC2)cc(N)cc(O)c1F C1(NC(c2cc(C)c(C)o2)=O)CCN(C(=O)COC2(C)CCCC2)CC1C C1(C)(CNC(C(c2csc(-c3ccccc3)c2)C)=O)CCCN(C(=O)C2CC2)C1 C1(N(C(c2cnn(C)c2)=O)CC)CCCN(C(c2cc(C)on2)=O)CC1 N1(CC(N2CCCCC2CO)=O)CCN(C(=O)Cn2cccn2)CC1 CC1CC2(CCO1)CC2C(=O)NCC(C1CCCN1c1nc(=O)n(C)[nH]1)(C)C c1(OCC(=O)NC2CC(NC(C3(COC)CCC3)=O)C2)cccc(Cl)c1.SCC N1(C(C(C)(C)OCCC)=O)CCC(CNC(C2(C)CC2)=O)C(CC)C1 C#CCC(O)C(=O)N1CCC(CCNC(=O)COCC(=O)OC)C1 CCC(COCCOCCN1CC=CC1)N=c1nc2c(cnn2C)c(NC)[nH]1 C1(CCNC(C2CC(OC)C2)=O)CC(F)(F)CN1C(c1csc(C#N)c1)=O c1(OC)cc(C=CC(=O)NC(C)CNC(c2c[nH]c(O)c2)=O)sn1 C1(CC(=O)NC2C(NC(CC3(OC)CC3)=O)CCC2)CCC2(CC1)CCC2O c1(C(N(C2CCOCC2)C(C)C)=O)ccc2c(c1)CC(=O)NC2 c1(C(=O)NCC23C(CN(C(C4N(C(C)=O)CCC4)=O)C2)C3)cc2c(ccn2C)s1 C(=O)(C(C)(C)C(C)(C)C)N1C(CNC(C2CC(OC)C(OC)C2)=O)CC2CC21 C1(C(=O)NC(CC)CN(C(c2ccccc2O)=O)CC)C(F)(F)C12CCC2 c1(C(N2C(C)CC(CNC(c3c(C)snn3)=O)C2)=O)cc2cc(F)ccc2s1 C1(CC(=O)N(C2(C(N(C)CCc3ncon3)=O)CCC2)C2CC2)C=NN(C)C1=O C(=O)(C#CC1CCCCC1)N1CCC(C(C)NC(CC(COC)(C)O)=O)CC1 CCCC(C(=O)NC1CC(C(=O)NCCc2cc(C)on2)C1)C(C)C CN1C(=O)CCC1C(=O)NCCCN1CCN(C(C2(F)C3CCCC23)=O)CC1 C1(CNc2cc(NC3(CCOCC)CCC3)ncn2)CCP(C)(=O)CC1 c1(C(N2CCC(NC(CC3(C=C)CC3)=O)CC2C)=O)cc(C)[nH]c(=NC)n1 CCN(CC(=O)NC)N1CCC(CCC(N)=O)CC1 C1(C(=O)NCC2C(C)(C)C(O)C2)CN(C(c2ccc(Cl)o2)=O)CC1(C)C CC1CCC(NC(C2CC(C3CC3)C2)=O)CN1C(c1cc(-c2ccco2)no1)=O c1(C(N2CC(NC(CS(CC)(=O)=O)=O)C(O)C2)=O)coc2cc(F)cc(F)c12 CCC(C)C(C(=O)N(C1CCC1)CCO)N(C(=O)CC1(C)CCOC1)C c1(C(=O)NC2C(C=C)C2)ccc(C(=O)NC(CSC)CN(C)C)cc1 c1(CN(C(=O)NCCOCCC=C)C)ccc(C)c(Br)c1 N1(C(c2c(C)c(Br)no2)=O)CC2(CCN(C(c3cocn3)=O)CC2)C1 c1(C(C(=O)NCc2ccccc2)N(C(C)CC(N)=O)C)ccc2c(c1)OCO2 C#CC(C(C)C)NC(=O)Cn1cc(CNC(=O)C=CCN2CCCC2)nn1 C12(CNC(COCc3ccc(C)cc3)=O)CN(C(=O)C(C)(Cl)Cl)CC1CCO2 c1(C(=O)NC2CC(N(C(C(CC3CC3)OC)=O)C)C2)cc(C(C)=O)cnn1 C1(NC(c2c(C)onc2Br)=O)CN(C(=O)CC(C)CF)C2(CCC2)C1 c1(C(=O)NCCCCC2CN(C(=O)CSn3cncn3)C2)nc[nH]c1C(F)(F)F C1(NC(c2ccoc2C(F)(F)F)=O)CCN(C(c2cccc(F)c2Cl)=O)CC1O Cc1cccc(C)c1OCC(=O)N(C(C)CNC(C1CCC(=O)CC1C)=O)C N1(C(C(CC)O)=O)C(CC(=O)Nc2ccc(C(N)=O)c(F)c2)C2CCCC12 C=CCC(Cc1ccccc1)C(=O)N1CC(N(C)C(C2CCS2(=O)=O)=O)C(O)C1 Cc1c(NCc2ccc(F)c(Br)c2F)nc[nH]c1=NCC1(C)CC2(CC2)C1 c1(CC)c(C(=O)NC(C)CN2CCCCC2)cnn1C.C12(CC1)C(=O)NC2.OCC c1(CC)ccc(CC(=O)N(C(C)CNC(C2CCCN(S(C)(=O)=O)C2)=O)C)cc1 C1(OCC)(CNC(=O)C(C)O)CN(C(c2ocnc2C2CC2)=O)C1 c1(C(N(C)CC2COCCN2C(=O)CC23CCCC2C3)=O)ncnc(O)c1F Cc1cc2c(C(=O)NC3CN(C(C4(C)CCNC4=O)=O)C3)nccn2n1 C12CCN(CC1)C2=O.n1(C(C(=O)NC2C(C)(CC)C2)C)cc(C(=O)OC)nn1 O=C(C1=Cc2ccccc2OC=C1)NC12CCCC1N(C(=O)C1=CCC1)CC2 C(C(CCC)C(=O)N(C)Cc1cc(CC)no1)NC(C1(CC#C)CCCCC1)=O N1(C(c2c(C)nccn2)=O)CCCC2(CCN(Cc3c(O)cccc3F)C2)C1 CN1CCN(C(c2ccc(C3CC3)cn2)=O)C(C(=O)NCc2cc(CO)no2)C1 C(=O)(C1=CCSC1)N1CC(CNC(C2CC(n3cc(C(=O)OC)nn3)C2)=O)C1 C(CCC(O)CO)NC(CCN(CC=C)C(C1CCC2(CC2)C1)=O)=O CCCC(C(=O)N(C1CC1)CC1CCN(C(C2CSCCS2)=O)CC1)OC CCC(C)CC(=O)N(C)CCN1CCN(C(=O)CCCc2ccccn2)CC1 c1(OC)ncnc(OC)c1NC(C1(C#N)CCN(C(c2cccnc2Cl)=O)C1)=O c1(NC(C(C)OC(c2cnn(C(CC)CC)c2C)=O)=O)ccc2nc(S)[nH]c2c1 CC1C(NC(c2cc(Cl)ccn2)=O)CCCN1C(c1ncc(Cl)nc1Cl)=O CC1CCC(S)CC1.c12ccccc1-c1cn(nn1)NC(=O)C1CC21.C1(F)CC1 C1(C(=O)NC(C2CN(C(C3CCC(CO)CC3)=O)CCO2)C)CCCCCC1 C1(N(C2COC(C)C2)C(C)=O)CCCCN(C(=O)CN2CCCNC2=O)C1 C1(C(=O)NC2CC3CC(NC(C(C)(C)OC)=O)C2C3)CCc2nnnn2C1 CC(C)CC(C(=O)N(C)C(c1cnn(C)c1)C)ONC(=O)C1(F)CCC1 c1(C(N2C(C)CC(CNC(=O)CSCC3CCCCO3)C2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(C(C)N(C)C)=O)C2CCCC1CN(C(c1cc(Cl)cc3c1CCC3)=O)C2 N1(C(CN2CCN(Cc3c(OC)cccc3Br)CC2=O)=O)C2CCC1CN(C)C2 c1(C(=O)NC2C3CN(Cc4cccc(O)c4Cl)CC23)cc(F)c(Br)cc1F CC1=C(C(=O)N2CCC(C)C(NC(=O)C=Cc3cnc[nH]3)C2)CCCO1 C1(C(N2CCC(C)(NC(CC(C)(C)N(C)C)=O)C2)=O)CCOC(C)(C)C1 C(C(C)(C)CC(=O)N(CC(C)O)CCNC(c1cnccc1C)=O)OC(C)=O N1(C(C(C)NS(CC)(=O)=O)=O)C2CCC1C(CNC(=O)CC(C)O)C2 C1(N(C(C(C=CC)O)=O)C)CN(C(c2cn3ccsc3n2)=O)CC1(C)C CC1CCCn2cc(C(=O)NC3CCCC3CNC(=O)CCOCC3CC3)nc21 CCCC(CCCO)C(=O)NCC1(C)CCN(C(C23CCCN(CCC2)C3)=O)C1 CCCCC(CC)CC(=O)N1CC(C)CN(C(c2nncs2)=O)CC1C c1(C(=O)NC2CN(C(CCCC)=O)CC(O)CC2)cc(S(=O)(=O)CC)cnc1O N1(C(=O)NCCCOC)CCC(C)(NC(C2CC(OC)C2)=O)C1 C=C=C(C)CC(=O)NCc1cccc(CCCCC)c1.C12CCN1NC2=O c1(OC)ccc(F)c(C(=O)NCCC(N)=O)c1Cl C1(NC(CCC(=C)C)=O)CC(F)CN(C(C2(CCC)CCNC2=O)=O)C1 CC1CN(C(c2cc(C(N)=O)[nH]n2)=O)CCC1NC(c1ccc(F)s1)=O n1(C(C)C)nc(C2CC2)cc1C(=O)NCC1(O)CC(NC(=O)C(C)O)C1 C1(NC(c2ccc(C(C)=O)o2)=O)CCC(C)N(C(C23CSCC2C3)=O)C1 C(C)(CC#C)(C(=O)NC(C)CCCO)NC(c1c(C#C)c[nH]n1)=O C=CCC(CC)C(=O)NC(C)(CNC(=O)Cc1ccn(CC)n1)C1CC1 N1(C(c2cc(C)ns2)=O)CCN(C(=O)CCc2nc(N(C)C)no2)C(C2CC2)C1 CCC(CCC(=O)N1CCCC1(C)C(=O)N(CCCN1CCCC1)C)OC C12(C(=O)Nc3cc(C)c(F)cc3)CCCC1CN(Cc1cc3n(n1)CCC3)C2 C12(C(=O)NCC(=C)CCNC(c3ccc(CN4CCCC4)[nH]3)=O)CCC(CC1)C2 c1(CNC(C2(OC)CCOC2)=O)ncc(C(=O)NCC2CCC2(F)F)cn1 c1(N(C)C(C2CCCN(Cc3cccc(Br)n3)C2)=O)ccc(I)c2cccnc12 N1(C(c2cccc(N(C)C)c2)=O)CC2C3CCC(C3)C2C1 Cc1ccc(CNC(=O)CCOCCNC(C2CCN(C)C2)=O)c(F)c1 C(=O)(C(CNC(=O)C(C(C)C)OCC)C(C)(C)C)NC(CCCC)CO C1(C(=O)NC2(CNC(CCOCC)=O)CCCCC2C)(CC)CCC(F)(F)CC1 C1(C(=O)NCC(C)(C2CC2)NC(c2ccc(C3CCC3)cc2)=O)CCC(C)CC1 c1(OC)cc(Cl)nc(CS(C)(=O)=O)n1.C12C3CN(CC13)C(=O)CN2 N1(C(c2cc(C)c(C)o2)=O)CCC2(COC(CNC(C3CC3C)=O)C2)C1 Cc1ccc(C=CC(=O)NC2CC2NC(=O)C=Cc2ccc(O)cc2)c(C)c1 c1(OC)cc(Cl)ccc1C(N1CC(OCCNC(C23CCC2CC3)=O)C1)=O C12(C(=O)OC)CCOCC1CN(C(=O)CC1CCN1C(c1cc(O)ncn1)=O)C2 C#CC1CN(C(=O)COC(F)(F)F)CCN1C(=O)C(F)=CCC CC1(C)CC(CNC(=O)CC(C)(C)NC(c2cnn(CCF)c2)=O)CO1 c1(NC(C(=O)NCC(CC(C)C)NC(=O)OCC)=O)cc2c(s1)CCCCC2 c1(OC)ccc2c(c1)CC(NS(=O)(=O)c1c(C)cc(C)cc1C)CC2 N1(C(Cn2nc(C)oc2=O)=O)CCN(C(=O)C=CCn2cncn2)C(C(F)F)C1 C1(C(=O)NCCCC)CCN(C(=O)CCc2ncc(C)[nH]2)C(C)C1 c1(CNC(C2C(CNC(Cn3ccc(C)c3)=O)CCO2)=O)ncccc1C CCCS(=O)(=O)CC(=O)NC1CC1CNC(c1cnn(CC2CCC2)c1)=O CCC(C)C(CN(C(=O)CCC1(C)CCCN1C(=O)C1=C(Cl)CC1)CC)CO C1(C(=O)NC(C2(O)CN(C(CNC(=O)OCC)=O)C2)C)CC2CCC1C2 C(C)(C)(CC(=O)NCC1(C)CC(NC(=O)CC2CCOC2=O)C1)SC C1(CCCNC(CCN(CCC)C)=O)CCCCN1C(c1nccn1C)=O CC1N(C(=O)CC2CCCC2NC(=O)CCN2CCCC2=O)CCCC1(C)C CCC(CC)CCC(=O)NC1CCCC(NC(c2cc(O)ncc2F)=O)C1 N1(C(C(CC)(C)CO)=O)CCCC(C2CN(C(C3(C#N)CCCCC3)=O)C2)C1 N1(C(C(N2CCC(C)C2)=O)=O)CC2CCC(CNC(=O)CC3(CO)CC3)(C2)C1 N1(CC(=O)NCC(CC)NC(c2cscc2C(N)=O)=O)CCCC1CC c1(CCC(=O)NCC(CNC(CCSC)=O)F)cnc2n1CCOC2 c1(CN(CCn2c(-c3ccc(CCC)s3)ncc2)C)ccc2c(c1)C(=O)CCC2 n1(CC(N2CC(NC(Cc3c(C)non3)=O)C(C)C2)=O)ccc2c(C)cccc12 Cc1nc(=N)[nH]c(=NCC2(C)CCN(C(C3(C)CCCCC3)=O)C2)[nH]1 C1(CCC(=O)NCC(C2CC2)C2CC2)CCCCN1C(=O)COCC1CC1 CC1(C)CN(C(=O)CC2CCCCCCC2)CC1CNC(c1coc(CO)c1)=O C1(OC(C)=O)CCCN(C(C)=O)CC1.O1P(=O)(OC2CC2)Cc2ccc(cc2)C1 Cc1nc(CNC(C2(CNC(=O)CCOCC(C)C)CC=CC2)=O)oc1C c1(CN=[N+]=[N-])cc(C(=O)NCC2OCCC2C(=O)NOCCN(C)C)n[nH]1 Cc1cncc2cc(C(=O)NC(CNC(c3cnc(C(C)C)[nH]3)=O)C(C)C)sc12 c1(C(N2CC(C)C(NC(=O)COC(F)F)C2)=O)c(OC(F)(F)F)ccc(F)c1N CN1CCC(NC(C2C=CCN2C(C2CCCCO2)=O)=O)C(C#N)C1 C1(CCOC)CN(C(C2(F)CC2)=O)CCN1C(C1CCN(S(=O)(=O)C(F)F)C1)=O C=CC(CC)CC(=O)NCC(O)C(=O)NCCN1CC2CC2C1 CC(C(=O)NCC1(NC(c2n[nH]c3ccc(O)cc23)=O)CC1)C(C)S(C)(=O)=O N1(C(C2(SCC)CCC2)=O)CCCC(CO)C1.C1(=O)C(COC)N1 c1(C(=O)NC2CCC(C(=O)NC(C3CCOCC3)C)C2)cc(Br)ccc1Br c1(OC)ccc(C(=O)NCC2(CCNC(=O)CCNC(C3(Cl)CC3)=O)CC2)nc1 C1(CNC(C(c2ccc(OC)cc2)C)=O)CC2(CCCN(c3nnc(C)o3)C2)C1 CC1=C(C(=O)NC2CC(N(C)C(c3cc4ccc(F)cc4o3)=O)C2)CCS1(=O)=O C1(c2ccc(C)cc2)C(C)CCCN1C(c1cn(CC(F)F)cn1)=O c1(C2(C(=O)NCC#CCNC(C3C(C)OCC3)=O)CCC2)ccc(Br)cc1 Cc1oc(C(=O)NCCC2CCCN(C(=O)CC3CCCCC3O)C2)cc1CO Cc1cnn(C)c1CC(=O)NC1CN(C)C(=O)O1.C1(CC)CC1CNC(=O)C1CC1 C1(NC(c2cc(CC)on2)=O)CCN(C(c2cocc2C)=O)CC1CO N1(C(COCCOC)=O)CC(n2cc(C(O)CC(C)C)nn2)C(C)C1 C1(C(N(C(CN(C(C2C(C(C)=O)C2(C)C)=O)C)C)C)=O)CCCCC1(C)C c1(C(=O)NC2CN(C(COC)=O)CC(C)C2)ccc(P(C)(C)=O)s1 C1(NC(CN(C(=O)NCCN2CCNC2=O)CC)=O)CCN(C)C1=O c1(NC(c2c(NC(c3cc(C)[nH]c3)=O)ccs2)=O)cn2c(N)cccc2n1.C(N)=O n1(CC)nc(C)c(C(=O)NC(C)CC(C)NC(c2cnccc2Cl)=O)c1C c1(OC)ccc(C)cc1C(=O)NCC1(O)CC(CNC(=O)CC(C)F)C1 c1(C(=O)NC2CC(NC(c3cc(C#N)[nH]c3)=O)C2)c(F)ccc2n[nH]cc12 c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)(C)C2CC2)ccc(C#N)c(O)c1 N1(C(CSCC)=O)CCC(O)(N(C(=O)CSc2cccnc2)CC2CC2)CC1 N1(C(Cc2ccc(C)o2)=O)CC(NC(=O)CC2CSC2)C(c2ccccc2)C1 N1(CC(=O)NCCCCNC(C(N2CCC(C)C2)=O)=O)C(=O)NC(C)(C)C1=O c1(C(=O)NC(C)CNC(c2cccc(C(F)F)c2)=O)cc2ncccc2[nH]1 C1(NC(C(c2c(C)nn(C)c2C)C)=O)CC2CN(C(c3csc(Cl)c3)=O)CC2C1 CC(C)CC(C)C(c1nnnn1CCCF)NCC1(CO)CC2(CCC2)C1 C#Cc1cccc(C(=O)NC2CCC(NC(c3ccc(CSC)cc3)=O)CC2)c1 c1(C(=O)NC2CCCCC2NC(c2coc(O)n2)=O)cnc2c(c1)NCC2 c1(C(=O)NC(C(C)NC(Cc2c(C)nsc2)=O)CO)c(C)nn(CCO)c1C C(C1CCCO1)=CC(=O)N(CCC)CCNC(=O)CCn1cnnn1 c1(CC)ccc(C(=O)NC(C2CCN(C(=O)C(C)OC)CC2)C(C)C)nc1 CC1COCCC1NC(c1c[nH]nc1CNC(c1cc(CO)on1)=O)=O N1(C(c2c(N)nccn2)=O)C2CCC1CC(C(N1CCCCC1C(N)=O)=O)C2 C(=O)(CCCC(C)NC(c1cc(CO)[nH]n1)=O)N(CCC=C)CC N1(CC(=O)N(C)CCNC(=O)CSCC2CCCO2)C(=O)CN(C)C1=O c1(C(=O)NCC2CCN2CC2CC=CCO2)ccc(C2CC2)cc1F c1(CCNC(CC2N(C(C(COC)O)=O)CCC2)=O)ccccc1C C1(CNC(C2C(C)CN(C(C3(C(=O)NCCO)CC3)=O)C2)=O)CCS(=O)(=O)CC1 C(C)(C(=O)N1CCC(CN(C)C(c2c(O)cccc2F)=O)C1)(C(C)C)NC(C)=O C12(NC(c3n(C)ccc3)=O)CC1CN(C(=O)Cc1ccc(C(F)(F)F)cc1)C2 CC1CCN(C(C2CC3(CC3)C2)=O)C1CNC(=O)CCF C1(C(=O)NC2C(CNC(C(=O)Nc3ccc(C)cc3)=O)C2)CN2CCN1CC2C C(=O)(C1=CC2CCCC12)NCC1(C)CCN(C(c2coc3c2CSC3)=O)C1 N1(C(COCC)=O)CCC(C)(C)C(NC(=O)CC(C)(C)c2cccs2)C1 c1(-c2ccc(CCCC)s2)ccn2nc(C(=O)Nc3sccc3CO)cc2c1 C(=O)(C(C)(F)C(=O)NC1CN(C(=O)C(c2ccc(N(C)C)cc2)C)CC1C)OC O=C(C1CCCc2nccn21)NC1CN(C(=O)Cc2cc[nH]c(=N)c2)C1 n1(CC)nnc2cc(C(=O)NCC=CCNC(C3CC3CC3CC3)=O)ccc12 N1(C(C2CCC(C)N2C(c2ccn(C(F)F)n2)=O)=O)CCNC(=O)CC1C CC1C2CN(C(=O)C(O)CNC(C3CC4(CC4)C3)=O)CC12 c1(C(=O)NCCOCCC)conc1CNC(c1ocnc1C)=O C(=O)(C1Cc2ccc(F)cc21)NC(CCCCNC(C1(C)C(CC)CCC1)=O)C c1(CC(C)C(=O)NC2CCC2NC(c2nnn(C)n2)=O)ccc(F)cc1 CN1CCN(C(C2CN(C(C3CCCC(=O)C3)=O)CC2(F)F)=O)CC1=O N1(C(C(C)OC)=O)CCC(C)(CNC(C2(C)CC=CCC2)=O)C1 C(=O)(C1=NN(CC)C(=O)CC1)NC1CN(C(CNC(CC)=O)=O)CC12CCC2 CC1(C)CC(C(=O)N2CCCC(CNC(=O)CN3CC4C=CC3C4)CC2)=NO1 c1(C(=O)NC(CCOC)CNC(C2CCSCC2)=O)cccc(C(C)=O)c1 C(CC(=O)N1CC(NC(C2(CC)CCCO2)=O)CCC1C)(C1=CCCC1)OCC C(=O)(C(CC(C)CC)NC(C1SCC=C1C)=O)N1CCC(CCC#C)CC1 CC1CC(CNC(c2ccnn2C2CC2)=O)CN(C(C2CCC3(CCC3)C2)=O)C1 Cc1cnoc1C(=O)NCC1C=CC(NC(C2(C)CCCO2)=O)C1 C1(NC(c2c(SC)scc2)=O)COC2CN(C(C3CCC(F)(F)CO3)=O)CC12 C1(CN(C)C)CCCN1C(=O)CC1CCCN1C(c1csc(-c2ncc[nH]2)n1)=O c1(C(c2nnnn2CC(F)F)NCC(c2cccc(C)c2)OC)noc(C)c1Br c1(C(=O)NC(C)CN(C(=O)CCN2CCOC2=O)C)cc2cc(Cl)ccc2s1 CC1CC(=O)N(C)c2ccc(C(N3CCC(O)C34CCSC4)=O)cc21 N=c1[nH]c(=NCc2c[nH]c3c(F)cccc23)[nH]c(=NC2CCCC2C#N)[nH]1 CC1(C)CCC(CC(=O)NC2CC(CNC(c3cnc(C(F)F)nc3)=O)C2)O1 N1(C(CN(C(=O)OC)C)=O)CCC(C(C)CNC(C2CC2(C)C(F)F)=O)CC1 C1(CC(=O)NCCC2CCC(NC(CSC(C)C)=O)C2)COC(C)(C)CO1 c1(C(=O)NCCC(C)N(C(=O)Cn2nccn2)C)csc(Cl)c1Cl Cc1cc(N)cnc1C(=O)NCC(O)CN(C(=O)C(C(C)(C)C)NS(C)(=O)=O)C C1(CNC(c2ccc(F)cc2Cl)=O)CCN(c2nnc(C3CC3)s2)CCC1(F)F C(=O)(CCCCSC)NC.C1(OC)(N)CN(C(C2(n3cnnn3)CC2)=O)C1 CC(CC(=O)N1CCC(CNC(c2ccc(-c3ccsc3)cc2)=O)C1)C(C)(C)C C1(C(=O)NCC2CC(NC(C(CCCC)C)=O)C2)CCc2nncn2C1 O=C(CC1OCCc2ccsc21)NC1CCN(c2nnco2)CC12CCC2 c1(CC(=O)NC2(CNC(C(CC=C)C(C)C)=O)CCC2)ccc([N+](=O)[O-])c(N)c1 C1(c2nc(CCC)nn2-c2cnn(C)c2)Cc2cc(C)ccc2S1 CC1CCc2ncccc2N1S(=O)(=O)c1cccc(Br)c1-c1ccc(F)cc1 Cc1c(C(N2CCC(C)C2C(N2CCCC2Cl)=O)=O)cccc1N c1(C(N(CCCN(CC(N2CCCC2)=O)C)C)=O)cn2ccc(Cl)cc2n1 C1(CCNC(C2(C)CC2)=O)CCCN(C(C2CCC(C)CC2)=O)CC1 C(=O)(CCCCC(C)C)NCCCCCC(=O)NC(C(=O)OCC)CO N1(C(C(C)CF)=O)CCCN(C(c2ccc(SC(F)(F)F)cc2)=O)CCC1 C1(C(=O)NCCCOC2CCC2)CC2(CCN1C(c1ccccc1)=O)CC2 c12ncnc(c1F)NC1CCC(C1)NC2=O.c1(CC)ccc(OC)cc1 c1(OC)ccc(Cn2nccc2-c2nc(C3CCCC3)nn2C2CCC2)cc1 C1(CNC(c2c(N(C)C)scn2)=O)C2CN(C(c3cn(CC4CC4)nn3)=O)CC12 C(c1ccc(Cl)s1)=CC(=O)NC1(CCCNC(C(C2CCOCC2)OC)=O)CC1 C=C1Cn2c(C(=O)NCCC(C)NC(C3OCCOC3C(F)(F)F)=O)nnc2S1 N(C)(S(N)(=O)=O)CC(=O)NC1CC(N(C(=O)CCC2CCCCC2)C)C1 N1(C(C(c2cccs2)N(C)C)=O)CC(CNC(=O)Cc2cc[nH]n2)C2(CC2)C1 C1(OC2CCC3(C(=O)NC(C)C(C)C(=O)N(C)C)C2C3)CC(C)N(C)CC1C N1(C(C2N(C)CCCC2)=O)CCCC(C)(C)C1CNC(c1ccoc1C1CC1)=O c1(C(C(=O)NCSc2ccccc2)N(C(C#C)C)C)ccnc(OCC)n1 C(=O)(CCS(N)(=O)=O)NC(CN(C(c1cc(OC)cc(Cl)c1)=O)CC)C C=CC(C)(CC)C(=O)N1CCC(N(C(=O)COC2CCCCC2C)CCO)CC1 N1(C(c2ccc(F)cc2)=O)CCC2CC12C(=O)NCCN1CCCCC1=O CCCCC(O)C(C)C(=O)NC1C=CCN(C(c2ccc(C)c(C#N)c2)=O)C1 C1(CCC(=O)N(C)CC2(C#N)CCC2)CCCCN1C(c1cocn1)=O C1(C(=O)NCCCCNC(C2OCCC2c2cnn(C)c2)=O)(COC)CC1(F)F C1(NC(c2cc(C(C)=O)cn2C)=O)CC(F)CN(C(=O)CC(C)(C)C)C1 C1(NC(=O)C=CBr)CCCC1C(=O)NCC1(F)CC1c1ccccc1 C1(C(C)N)CCCCCC1.C(C(C)(C)C)(c1nnnn1CC(F)F)CCC1(C)CC1 C1(CCC)(C(=O)NC(C)CN(C(=O)CSc2ccncc2)C)CCNC1=O c1(OC)ccc(Cl)cc1CC(=O)NCCC1CCCN(C(=O)COC)C1 N1(C(C(CCC)CC)=O)CC2(CCN(C(c3cccc(C)c3Cl)=O)C2)C1 C(C(C)C(=O)NC(C(F)(F)F)C1CC1)NC(C(C)NC(=O)C1CC1)=O CC(C)C#CC(=O)N1CC=CC1CNC(=O)C(c1ccccc1)C CC1CCc2[nH]c(=NC(C)c3cccs3)nc(N3CCc4cnn(C)c4C3)c2C1 c1(OC)cc(C(N2CC3CC2CN3C(=O)C=Cc2sccc2C)=O)cc(C)c1 c1(C(=O)NCC(CNC(=O)CCN2CCOCC2)OC)nccc(N)c1Cl CCC(CC)CCCC(=O)N(CCCN(C(=O)CN(C)C(C)=O)CC)C c1(C(=O)NCC(CC(=O)N2C(C(C)C)CC2)(C)C)cnn2ccc(Cl)c(F)c12 N1(CC(=O)NC2C(CNC(=O)Cn3nccc3C(F)(F)F)C2)CSCCSC1 Cc1ccn2cc(C(=O)N(CC(C)NC(C3CC34CCCCC4)=O)C)nc2c1 C=CC1(C(=O)NCCC(C2CC2)C2CC2)CCN(C(C2CC23CC3)=O)CC1 C1(NC(c2oc(CC)c(C)c2)=O)CCN(C(c2ncc(OC)cn2)=O)CC(O)C1 C1(NC(C(C)=CC2CC2)=O)CCN(C)C12CCCN(C(=O)Cc1n[nH]c(=N)s1)C2 CN1CC(O)CC1(C)C(=O)NCC1CCN(C(=O)Cc2cscn2)CC1 c1(C(N(C2CCN(C(=O)CC=C(C)C)C2)CCC)=O)ccc2c(c1)CCN2C c1(SCC)nccnc1C(=O)NCC1(NC(C2CC(=O)OC2C)=O)CCOC1 Cc1cc(C(N2CCCC2CN(C(=O)C(Cl)(Cl)Cl)C)=O)nc2nccn12 N1(Cc2cc(C)[nH]c2)CCC(Cc2cc(-c3ncccc3O)n[nH]2)CC1 c1(C(CC)CC)nc(-c2nnn(CC)c2N)n(-c2ccn(C)n2)n1 c1(C(=O)NC2CC3(CN(C(c4scc(C)c4)=O)C3)C2)c(C)[nH]c2ccc(F)cc12 C1(CNC(CC2N(C(C(C)(C)c3cccs3)=O)CC2)=O)CCCC12CCC2 C#Cc1ccnc(C(=O)NCC23CC(C2)C(NC(=O)CSC2CCCC2)CO3)c1 N1(C(c2c(N)cccn2)=O)C2CCC1C(C(=O)NCCCN1CCOCC1)C2 C1(CC)C(C(=O)NCC2CCOC2C)CCCN1C(C1CCC(F)CC1)=O C1(O)(CCOCC)CCCN(C(=O)CNC(=O)CNC(C2(C)CC2)=O)C1 N1(C(C2C(C)N(C(c3cnns3)=O)CCC2)=O)CCC2CCN(C)CC12 Cc1nc(CNC(=O)CC2CCCN2C(=O)C(C)(C)CCl)sc1I C1(OC)CC2CCC(C1)N2C(C12CC(CN1C(C1CCCSC1)=O)C2)=O C12(CNC(=O)Cc3csnn3)CN(C(C3CCNC3=O)=O)CC1CCO2 C(C1CCOCC1)=CC(=O)N(CC(CC)NC(C1CN(C)C(=O)N1)=O)CC C1(OC)CCOCC1NC(=O)C(O)CCNC(=O)C(C)C1CC1 N1(C(C(N(C)C)C2CC2)=O)CC(NC(c2ccc[nH]2)=O)C2(CCOCC2)C1 C=C(CNC(=O)CCC1CCC(C)O1)CCNC(C12CC(CC(F)F)(C1)C2)=O C=C1CN2C(=O)CCC2(C(=O)NC2CCC(NC(=O)Cn3ccc(C)n3)CC2)C1 N1(C(c2cc(OC)ncc2)=O)CCC(CO)(CNC(C2C3CCCC23)=O)CC1 c1(C(=O)NC(C)CCNC(C2CN3CCN2CC3)=O)csc(S(C)(=O)=O)c1 C(CCNC(=O)C(Br)=C(C)C)(C(C)(C)C)NC(C=C(CC)C)=O C1(NC(CCNC(C)=O)=O)CCCOC12CCN(C(C1CCC(C)O1)=O)CC2 C1(OCC(=O)NC(c2ccccc2)C)CCN(C(=O)COCC2CC2C)C1 C1(NC(c2c(C)nco2)=O)CCN(C(c2ccc(N(C)C)cn2)=O)CC12CCC2 CCCC(C(=O)NCC(C)CN(C)C(c1cc(OC)no1)=O)N(C)C C(=O)(CC(C)(O)C(F)(F)F)NC12CC(CNC(C3C(C(=O)OCC)C3)=O)(OC1)C2 C12(CNC(c3c(C)onc3)=O)CCC(CC1)N(C(C1CCCCC1(C)C)=O)C2 c1(C(c2n(CCCC)nnn2)NCc2cc(C)no2)ccncc1OCC Cc1ccc(CCC(N2CC(NC(c3nc(O)sc3C)=O)C(C)C2)=O)cc1 C1(NC(CCC#CC)=O)CC(CNC(=O)Cc2nc[nH]n2)C12CCC2 c1(C(=O)NC(CC)CNC(c2ccc(C(C)F)cc2)=O)noc2cc(F)ccc12 N1(C(C(N2CCCCCC2)C)=O)CCCC(c2cccc(C(=O)O)c2)C1 CCC(C(=O)N1CC(C(C)C)C1)NC(C1CC1Cl)=O Cn1cnc2[nH]c(=NCc3cscn3)nc(N3CCOC(C#N)C3)c12 CN1CCN(C)CC(C(=O)NC2CCCCC2NC(c2cnc(=N)[nH]c2)=O)C1 CCC(CO)CN=C(NCc1snnc1C)NCC1CCOC1 c1(C(=O)NC(C2CCC2)C)c[nH]c2ncc(-c3ccc(F)cc3F)cc12 N1(C(c2ccn(CC)n2)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(CC2CC2)C1 CC(C)C(CCNC(c1ccc(-c2cccnc2)s1)=O)NC(=O)C(O)C1CC1 c1(C(=O)NCC(C)NC(c2ccc(F)cc2Cl)=O)cccc2c1OCC2 N1(C(C(C)OCCOC)=O)CCC2CCC(NC(c3ncc(Cl)s3)=O)C1C2 c1(C(=O)NCCCN(C(=O)C(F)n2cccn2)C2CCCC2)cncnc1 C(c1ccc(C(=O)OC)cc1)=C(CN1CC(C=C)C1)C C1(CNC(c2ccoc2Cl)=O)CCCCN(C(c2cc(C3CC3)ccc2Cl)=O)C1 c1(C(C)=O)ccc(O)c(C(=O)NCC2C3CN(C(c4cn(C)cn4)=O)CC23)c1 N1(C(CCc2ccc(C)s2)=O)CCC(C)C(NC(=O)CCN2CCCS2(=O)=O)C1 c1(OC)oc(C)nc1C(=O)NCC(CC(C)C)NC(C1CCCO1)=O C#CCCCCC(=O)NC(Cc1ccccc1Br)C(=O)NC1CCN(C(N)=O)C1 C12(CC(=O)N(C(C)C)CCO)CCC(CC1)C2.c1(C2CC(=O)N2)cccc(Cl)c1 C1(NC(CC2(C#N)CC2)=O)CCCC(F)C1 C1(C(=O)NCC(Cc2ccccc2)NC(CCNC(C2C(C)C2)=O)=O)COC(C)C1 N(C1CCCc2c[nH]nc21)C(C1(NC(=O)CCc2nccs2)C(C)CCC1)=O c1(CC(=O)NC2CC(NC(C(CC=C)C)=O)C2)c(C)cc(C#N)cc1C N1(C(COCCC#C)=O)CC(C)(C)CCC1CNC(=O)COCC(=C)C CC(C)(O)C(C)(C)C(=O)N1CCCC(NC(c2cccnc2S)=O)C1 c1(C(N(CCNC(C2C(C=C)OCCC2)=O)CC)=O)cc(Br)cc(C)c1F CC1(NC(c2ccsc2)=O)CCN(C(=O)CC2CCOC2)CC1 C1(CNC(C(C)=CC2CC2)=O)COCCN1C(c1cnnn1-c1ccccc1)=O c1(C(=O)NC2C(NC(c3c(C(C)C)con3)=O)CCCC2)nsc2ccccc12 N1(C(C2(CCOC)CCCC2)=O)CCC(F)(CNC(C2(CC3CC3)CCC2)=O)C1 C1(C(=O)OCC)C2COC(C(=O)N(C)CC3CCN(C(=O)CC4(C)CC4)C3)CC12 C1(NC(C2(C(=O)NC)CCC2)=O)C2CN(C(=O)CC(c3c(C)noc3C)C)CC12 C1(NCCC(=O)NCC2CCN(C)C2)CCc2ncc(Br)n2C1 c1(C(=O)NCCCC2CN(C(c3ccc[nH]3)=O)CCO2)c[nH]c2ncnc(O)c12 N1(C(c2cc(C(=O)OC)ncc2)=O)CC2(CCN(C(=O)CCC(F)(F)F)C2)C1 CCC(C)(O)CCNC(C1C(C(=O)NC)CCO1)=O S(=O)(=O)(c1cc(N2CCCC3(CCc4ccccc43)C2)c(C)c(Cl)c1)NCCOC C(=O)(C1=CCOCC1)O.c1(CN(C(=O)CNS(C)(=O)=O)CC)csc(C)n1 N1(C(c2nc(NC(=O)C=CC3CCC3)sc2)=O)CCC2(N(CC)CC)CCCC12 c1(C(=O)NC2CC(NC(CCCCC#N)=O)C2)c(F)c(F)c(F)c(F)c1F Cc1nn(-c2ccccc2)c(NCCNC(c2c(O)ncnc2O)=O)c1[N+](=O)[O-] C1(C)(C(N2CC3C(CNC(CN(S(C)(=O)=O)C)=O)C3C2)=O)CC(=O)N(C)C1 c12cc(F)ccc1CNC2=O.C1(C)(C(=O)OC)CN(C2CC2)C1=O CCCC(O)CC(=O)NC1CC(NC(c2cc(NC)nc(Cl)c2)=O)C(O)C1 C(=O)(C(O)CC(F)(F)F)NCC12OCC(C(=O)Nc3c(F)cccc3F)(C1)C2 c1(NCC)ccc(C(=O)NC2CCCN(C(=O)CCCN=[N+]=[N-])C2)cc1[N+](=O)[O-] c1(C(=O)NCCCCNC(C(CC)N(C)C)=O)cnn(-c2ccccc2F)c1C N1(C(c2c(C)con2)=O)CCC2(CC1)CN(C(=O)CC(C)C(F)F)CCO2 c1(C(N2CCC(NC(c3[nH]cc(C(C)=O)c3)=O)C2C)=O)ncc(N)cc1Cl n1(CC(=O)NCC2C3CN(C(=O)C=C4CC4)CC23)ncccc1=O c1(C(N(CCOC)CCNC(=O)C(F)(F)C2(O)CCC2)=O)ncc(C#N)cc1Cl Cc1cc(=NCC2(N(C)C)CCSC2)[nH]c(=NCC(=O)N2CCCC2)[nH]1 c1(C(=O)NC(CC=C)CNC(=O)Cc2cc(C)n(C)n2)nc2ncc(C)cn2n1 c1(-c2ccc(NC(c3cc(Cl)nc(Cl)c3)=O)nc2)cnn2ccccc12 c1(C(C)C)cc(N2CC3CCC2C(NC(=O)CC(F)(F)F)C3)n2ncnc2n1 C12(CNC(c3c(CC)n[nH]c3)=O)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 S(=O)(=O)(c1ccc(C)cc1)NC(C(N1CC(COC)C(C(F)(F)F)C1)=O)C C(C1Cc2ccccc21)NC(c1c(CNC(c2c(C)ccc(C)n2)=O)ccs1)=O Cn1cc2c(n1)CC(C(N1CCC(C)(NC(=O)CN3CC(=O)NC3=O)C1)=O)CC2 C1(C(N2CCC(NC(CCCCC)=O)C(C)C2)=O)CCS(=O)(=O)C1(C)C c1(C(=O)NC2C(NC(CCOCCN(C)C)=O)CCCC2)csc2ccccc12 N1(C(c2cccc(CC)c2)=O)CCC(C)N(C(=O)C(CCSC)OC)CC1 CC1(C)CN(C(=O)C(N2CCOC(CC(N)=O)C2)=O)CC(CO)O1 c1(C(=O)NC(CNC(C(CC)(C)C#N)=O)C2CC2)cc2c(F)c(F)c(F)cc2[nH]1 C#CC1CCC(C(=O)NC2CCCC(CN(C)C(c3ccc[n+]([O-])c3)=O)C2)CC1 N1(C(CC(CC=C)(C)C)=O)CCC(NC(c2scc(Cl)c2Cl)=O)C(F)(F)CC1 C(=O)(C1=COCCC1)NC1(C)CC(NC(C2(C(F)F)CCCO2)=O)C1 C12(C(=O)NCc3c(OCCC)cccn3)CCC1CCN2C(=O)CCCSC N1(C(c2ccc(C)cc2Br)=O)CC(NC(=O)CC(C)N(C)C)CC2(CC2)C1 Cc1cc(Br)cc2c(NC(=O)N(C3CN(S(=O)(=O)C4CC4)C3)C)ccnc12 c1(C(C)NC(=O)Nc2c(C(=O)OC)[nH]c(C)c2)nc2ccccc2s1 N1(C(C(C)=CC)=O)CC2CCN(C(c3sc(Br)cc3F)=O)C2C1 c1(C(=O)NC2CC(N(C(=O)CN3CCCC3=O)C)C2)c[nH]c(=O)c2ccnn12 CC(CN=C(NCC1CC=CCC1)NC1CCCC1)Oc1ccccc1Br CC1CCN(C(=O)Nc2nccnc2Br)CC1N1CCCC1 C(CC(=O)NCCCN(CC1CC1)CC)SCCCC.N(S(N)(=O)=O)CC=O C(=O)(C1CCCc2scnc21)N1CCC(C(=O)OC)C12COC2 CCCC(C(O)C(=O)N1CCC(C#N)CC1)NC(=O)CC1CCSC1 C1(C(=O)NCCOCC=C)CN(C(c2cnc(COC)s2)=O)CCC1(C)C c1(NC2C(NC(c3ccc(C(C(C)C)=O)cn3)=O)C2)ncc(Br)cn1 CN=c1[nH]c(SC)ncc1C(N1CCC(O)C1C(=O)NC(C)COC)=O C1(CNC(C2(COC)CCCCO2)=O)C(C2CC2)CCN1C(=O)Cc1cnns1 N1(C(C(n2cc(-c3c(Cl)ccc(OC)c3)nn2)C)=O)CCC(O)C(C)(C)C1 C(CC(C)CC)(C(=O)N1CC(O)CC(C)(C)C1)NC(C1(CCCC)CC1)=O N1(C(c2ncc(CC)[nH]2)C(=O)NCC2CCCO2)CC(CO)OCC12CCC2 Cc1cncc(C(=O)NC2CC(CNC(=O)CCC3(C)N=N3)C2)c1Cl N1(C(C(CSC)O)=O)CC2CC1CC2CNC(c1n[nH]c(C)c1Cl)=O N1(C(Cc2ccc(C)cc2)=O)CC(F)(F)CC1C(=O)Nc1c[nH]nc1Br c1(-n2cc(CCN(C(=O)Cc3ccn(C)c3)C)nn2)cc(F)cc(F)c1 N1(C(CSCC#C)=O)CC(NC(=O)Cc2ccc(CCC)cc2)CC(C)C1 C1(CNC(C(C)O)=O)Cc2ccccc2CN1C(c1cc(Br)n[nH]1)=O C(=O)(C1=NOC2COCC12)N1CC(C)N(C(c2cc(N)cc(F)c2)=O)C(C)C1 Cc1cc(C)c(C(=O)NC2CC(N(C)C(c3cc(Cl)c[nH]3)=O)C2)cn1 c1(SC)cccc(CC(N2CC3CC3(CNC(=O)Cc3cc[nH]n3)C2)=O)c1 Cc1cc(CN(C)C(c2cn(CCNC(C3(C)CC3)=O)cn2)=O)on1 c1(NC(N(C(c2cccs2)C)C)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(CCC=C)=O)CC2(CCN(C(=O)CC3CC3)CC2)c2ccccc21 C(=O)(C(C)(C)n1cccn1)N1CC(CNC(C(C)NC(CC)=O)=O)C1 CC(C)C(F)C(=O)NCC(C(C)C)NC(c1ccccc1OCC#N)=O N1(C(c2cccc(Cl)c2Cl)=O)CCCN(C(C23CCN(CC2)C3)=O)CC1CO N1(C(c2cc(C)n(C(C)C)n2)=O)CC2CCC(C1)N2C(=O)CC1CC(C)(C)OC1=O c1(CC(N2C(CNC(c3cnc(CO)cn3)=O)CCC2)=O)ccc2c(c1)CCC2 N1(C(COC(C)C)=O)CCCC1C(C)NC(=O)Cn1ccnc1C(C)C c1(CO)c(C(=O)NCCC2(NC(=O)C(F)C3CCC3)CC2)sc2ccccc12 C#CCCCCC(=O)NC1COCCC1NC(=O)C(N1CCCCC1=O)C c1(C(=O)NC2C(NC(=O)CCc3cccs3)C2)ccc(-c2ccccn2)nc1O C1(NC(C)=O)CC2CCC(C1)N2C(c1sccc1Oc1ccccc1)=O C(C(C(=O)NC1C2CCCC1CC2)C(C)(C)C)NC(c1c(CC)c[nH]c1)=O C(N(C)N1CCC2(CC1)OCc1ccccc12)c1ccc(OC)cc1OC C(CCCNC(=O)CC1CC1CNC(=O)C(C)O)OC.C1(CN)CC1 Cc1ccncc1CC(N1CC(C)(NC(c2occc2Br)=O)C1)=O C1(NC(c2ccccc2[N+](=O)[O-])=O)CCC2CCN(C(c3sccc3F)=O)C12 C1(CNC(C(Br)=C(C)C)=O)CCC2(CN(C(C3OCC3(C)C)=O)C2)O1 O=C1CCCC(C(=O)NC2CC(O)(CNC(C3CCSCC3)=O)C2)O1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(CCNC(C(CSC)O)=O)CC1CC1 CC1CCn2ncc(C(=O)NCC(C)(C3CC3)NC(C3(C4CC4)CCC3)=O)c2C1 N1(C(c2scc(C)c2Cl)=O)CCC(C)(CNC(=O)CN2CC3CCC2C3)CC1 C1(C(N(C)CCN(C)C2CC2)=O)(NC(=O)CC2CC2(C)C)CCCCC1 c1(C(=O)NCC2CN(C(CN(C3CC3)CC)=O)C3C2C3)cc(F)cc([N+](=O)[O-])c1 C1(NC(=O)CSC2(CC(=O)Nc3cccs3)CCC2)CC2CC2C1 C1(=O)C(Cc2ccsc2)N1.C(=O)(CN(C(C)COC(C)C)C)NC(=O)OC C12(C(=O)NCCCN(C(=O)C(C)CC3CCCCC3)C(C)C)CCCC(C1)OC2 c1(CNC(CCC2N(C(C(n3c(C)ncc3)C)=O)CCC2)=O)cncc(Br)c1 C1(NC(C(N2C(c3cc(C)c(F)cc3)CCC2)=O)=O)CCCCCC1(F)F c1(C(=O)NC2CCCC(NC(CC3(C)CCCO3)=O)C2)cn2cnnc2cn1 CC1CCCC(C(=O)NCC(F)(F)Cn2cc(-c3cnccc3C(=O)O)nn2)C1 c1(C(=O)OC)cn(CC(=O)OC2(C(=O)OC)CC3C=CC2C3)n2ccnc12 c1(CN2CCCC(NC(c3ccc(Cl)c(Cl)c3)=O)CC2)c(F)cc(O)cc1F C1(C(N(C(CC(=O)NCc2nc(C)c(C)s2)C)C)=O)CC2(CCC2O)C1 C1(C(=O)NC2CN(C(C3(C(=O)OC)CC3C)=O)C2)CSCC(=O)N1 C12(C(N(CC(C)CNC(c3ccccc3C3CCC3)=O)C)=O)CC=CC(C1)OC2 c1(C(=O)NC(CC=CC)CO)cc(O)ccc1F C1(C(=O)NCC(C)CNC(c2ccc(Cl)nc2O)=O)C2CCC3(COC(=O)C13)O2 c1(OC)ccccc1C=CC(=O)NC1CCN(C(C2CCSCC2)=O)CC1F N1(C(CCC(=O)NCC)=O)CCOC(C)C1C(=O)Nc1ccc(F)cc1 c1(C(N2CCCC(C(=O)OC)CC2)=O)cc2c(C)cc(OC(F)F)cc2o1 N1(C(c2ccn3c(O)nnc3c2)=O)CCC2(CC1)CCN(c1cnc(F)cn1)C2 c1(CC(=O)NC)ccccc1C.n1(C(C(=O)NCC2CC(CC)C2)C)ccnc1C c1(CN2CCC(C)(NC(C(C)O)=O)CC2)cc(Br)c(F)cc1[N+](=O)[O-] C1(CC)CCN(C(=O)C=C2CCOCC2)C1CNC(=O)C(C)n1cncn1 N1(C(=O)NCCc2cc(OC)cc(Br)c2)CCC2(CCCCC2)C1C.C(COO)S c1(CN2CCC(C)(NC(c3cn[nH]c3)=O)C2)ccc(F)cc1C(=O)OCCO CC1ON=C(C(=O)NC2COCCN(C(C3(C(=O)N(C)C(C)C)CC3)=O)C2)C1C c1(C(=O)NCC2N(C(C(C)O)=O)CCC(C)C2)coc2cc(O)ccc12 C1(C(N2CCCC(C(C)C(=O)NCC(C)(O)C3CCC3)C2)=O)(OC)CCOCC1 N1(C(CC(C=C)C)=O)CCC2CN(C(c3[nH]cnc3CC)=O)CCC12 C1(c2scc(C(C)(C)C)n2)CCCN1N1CC(O)CC2(CCOCC2)C1 C1(C(=O)NCc2c(C(=O)O)nccc2)OCCOC12CCC2 N1(C(=O)NCC2C(C)(C)C3CCC2C3)CCC(=O)Nc2cc(F)ccc21 N1(C(C2CCC(=O)O2)=O)CCC2CCN(C(c3cccc4c3OCO4)=O)CC2C1 Cc1c(C(N2CCC(NC(C34CC(C)C3C4)=O)C2C)=O)nn(C)c1Br C1(O)(CCNC(c2c(SC)ccs2)=O)CCN(C(c2cscc2C(N)=O)=O)CC1 C#Cc1ccc(C(=O)NCC23CCC(CO2)C3)c(C)c1.C1(=O)CC(C)(C)C2CN1C2 N1(C(C2ON=C(C)C2)=O)C2CCC1CN(C(=O)CCc1cccn1C)C2 c1(OC)cnc(C(N2CCCC2(C)CNC(=O)CCc2ccn(C)n2)=O)cn1 C1(OC)CC2(CCC(C(=O)NCC3C4CN(C(=O)CC5(O)CCC5)CC34)CC2)C1 C1(CC)CCCCC1NC(c1n[nH]cc1CNC(=O)Cc1sccc1C)=O N1(C(CNS(C)(=O)=O)=O)CC2CC2(NC(c2ccccc2-c2cccnc2)=O)C1 C1(C(=O)NCC2CC(NC(c3c(F)ccc(OC)c3)=O)C2)CCC2C(C1)C2(F)F C1(C(=O)NC2CCC(CNC(C(COC)(F)F)=O)CC2)COc2ccccc2C1 c1(C(N2CCCC(CN(C(c3c(CC)cco3)=O)C)C2)=O)cc(C)c(F)cc1O C(=O)(C(CC(=C)C)OC)NC(CNC(CC(=C)C)=O)CCOC C#Cc1ccc(F)c(C(=O)NCCCCC(C)NC(=O)CC2(OCC)CCC2)c1 Cc1cnc(NC(C2CCCN(Cc3cnc(Cl)c(Cl)c3)C2)=O)c(C)c1 c1(C(=O)NC2C(NC(CC(=O)NC3CC3)=O)CC2)ccnc(F)c1F N1(C(c2cccc(OC)c2)=O)CCN(C(c2cc(Cl)ccc2O)=O)CC1C C(=O)(CC(C)(C)CC)NCCN(CCC)C(c1cc(Br)cn1C)=O c1(C(=O)NC2C(NC(C3(N(C)C)CCCC3)=O)CCC2)cccc2oncc12 CCC(F)(F)C(C)(C)C(=O)N1CC(N(C)CC)C1.c1(CCNC(=O)CO)ccccc1 N1(C(COCc2ccc(C)cc2)=O)CC2(CCN(C(c3cn(C)c(C)n3)=O)C2)C1 C1(NC(C2N(CC)CC2)=O)CCC(CNC(=O)C=Cc2cc(OC)ns2)CC1 C1(C(=O)NCC(C(C)C)(C)NC(=O)C(=C2CCCCC2)F)CN2CCN1C(C)C2 C1(NCCC(=O)N)CCCCN(C(=O)CC2(CO)CC2)C1.c1(C)ccccc1 c1(C(=O)NCC(CNC(C(C=C)(C)C)=O)OC)ccc([N+](=O)[O-])c(SCC)c1 CC1CCCC=C1C(=O)NC(c1cnn(C)c1)C(=O)N1CC(N2CCC2)C1 c1(CCC)ncc(C(=O)NCCC2(CNC(c3nnsc3C)=O)CC2)s1 C#CC1(CNC(C2(NC(c3cn(C4CC4)cn3)=O)CCSC2)=O)CCC1 C1(NC(c2n(CC=C)ccc2)=O)CN(C(c2cc(C(C)C)n(C)n2)=O)CC12CC2 N1(C(CC=C)=O)CCN(C(c2nc3cccnc3s2)=O)CC(O)C1 C(=O)(C1=NOCC1)NCC1(C)CC(NC(c2[nH]ccc2-c2ccccc2)=O)C1 c1(OCC)ccccc1.C(=O)(CCS)N(CCNC(CC1(OCC)CC1)=O)C C1(C)CCN2C1C2=O.C1(CC)CN(C(=O)O)C1.C(C)(C)(C)NC(=O)CC1CC1 C1(NC(C2CC(F)(CO)C2)=O)CCCCC1CNC(c1ncsc1C1CC1)=O O=C(N=c1ccnc(CNc2cc(Br)c(O)cc2Br)[nH]1)C1CC2CCC1C2 C(=O)(C(CC(C)(C)C)NC(=O)CC1CCN(C)C1=O)NCCC=C=C C1(CNC(c2occ(C)c2)=O)CC(C)N(C(=O)C(C)Cc2ccccc2)C1 N1(C(c2ccc(C(C)=O)o2)=O)C2CCC1CC(N(C)C(C1CCC13CC3)=O)C2 CC1(NC(c2nocc2Cl)=O)CCN(C(C2CCCOCC2)=O)C1 C=CCCCC(c1nnnn1CCCSC)NC1(c2ccc(CSC)cc2)CC1 Cc1cc2sc(C(=O)NCC3CN(C(c4cnc(O)o4)=O)C3)cc2s1 N1(C(C2(COC(C)C)CC2)=O)CCC2CCN(C(C3CC(C)(C)CCO3)=O)CC12 C(=O)(CCCC(=O)NCCN(C)C(c1ccn(-c2ccc(C)c(Cl)c2)n1)=O)OC N1(C(CC2(OC)CCOCC2)=O)CC2CCCN(C(=O)C(C#N)C3CC3)C2C1 C1(NC(CCOC(C)=O)=O)CCC(C)(NC(c2cnsn2)=O)CC1 c1(CC(C(=O)NCC2CC(NC(c3cnc(C)[nH]3)=O)C2)C)cccc(Cl)c1 C1(NC(CCOCCC)=O)CCC(NC(C2(CC3CC3)CC2)=O)CC1 C(c1ccc(C)s1)=CC(=O)NCCC1N(C(C2CC(OC(C)(C)C)C2)=O)CCC1 CC(=O)C(C)CC(C)C(=O)NC(c1cccnc1)C(=O)NCC(O)C(C)O c1(OC)noc(C)c1C(=O)NC1CC(CCNC(C2CNC(=O)O2)=O)C1 O=[N+]([O-])c1cccc(N2CCN(Cc3sc(I)cc3Br)CC2)c1 C1(NC(CSCC(=O)OC)=O)CN(C(=O)CC2CC2)CC1SC1CCCCO1 C1(NC(C(c2cnccn2)C)=O)CCCN(C(=O)COCCC2CCCC2)CC1 c1(NC(CNC(=O)NCC2CC(=C)C2)=O)ccc(OC)nc1 C(CNC(=O)Cc1nccn1C)(CC(=O)NOCCC1CC1)OC C(CCCCC(=O)NC1CCCCC1(C)O)N(C(C1CCC(CC)O1)=O)C c1(CCCC)cccc(C(=O)NCC2C(C)CCN2C(=O)C=[SH]C2CCCC2)n1 C1(C)(SC)CN(C(C2COCC2NC(=O)COc2ccncc2)=O)C1 C1(NC(C(n2ccc(C3CC3)n2)C)=O)CCN(C(=O)Cn2cccnc2=O)C1C CCCCC(CC(=O)N(C)C(c1ncccn1)C)NC(=O)C(C)CC N1(C(CCc2n(C)ncc2)=O)CCC2(CCCN2C(C2CSCCS2)=O)C1 C1(NC(C=CCN(C)CC)=O)CCC2CCN(C(c3nccc(OC)n3)=O)C1C2 CC(C1=Cc2ccccc2OC1)N1CC(O)CC1CC(C1CCCO1)O N1(C(CC(CC)O)=O)CC2(C1)CN(Cc1cncc(O)c1)C2 C1(Nc2cc(N3CCC(O)C3)ncn2)(CO)CC2CCCC2C1 C(=O)(C(CC)CC(C)C)NCCC(C)(C)NC(c1c(CC)ocn1)=O C1(CN2CCCC(NC(=O)CS(=O)(=O)NS(=O)(=O)C(C)C)C2)CCC2(CCC2)C1 N1(S(=O)(=O)CCn2nccn2)CC2(CCC2)C1C1CCCO1 CCC(CC(=O)NCC1CC(N(C)C)C1)NC(=O)CC1(C#N)CCC1 C1(C)(C(=O)NCC2(O)CN(C(c3c(C)onc3)=O)C2)CC2CCC(C1)S2 N1(C(C2C(C(C)NC(C(CC)OC)=O)C2)=O)CC(F)(F)C1C1CC1 C1(CNC(=O)Cc2ccc(CO)cc2)CC2CCC(C1)N2CCn1ncnn1 Cc1ccc(C)c(C(=O)NCC(C)(C(C)C)NC(C2CCCC2C(C)C)=O)c1N Cn1nnc2c1CC(C(=O)NCCOCCNC(c1ncc(Cl)cc1F)=O)CC2 c1(C(N2CCN(C(c3nocc3Cl)=O)C3CCC23)=O)ccc(Cl)c2ncccc12 C#Cc1ccnc(C(=O)NCc2nocc2C(=O)NC2CC2C)c1 N1(C(CC2(COC)CC2)=O)CCC(SNCCC(=O)NC(C)C(C)CC)CC1 C1(CCC#C)CCCN1C(=O)C=CCC(C)(C)NC(=O)C(F)C1CCCC1 C(CCCC(C)NC(=O)CC(C)CN(C)C)NC(C(C)CC1CCC1)=O C1(NC(C2CCC(N(C)C)CC2)=O)CCN(Cc2cn(C(C)C)nn2)C(C)C1 C12(NC(CC(COC)C)=O)CCC(C1)N(C(c1ccc(N3CCCC3)cc1)=O)C2 Cc1c(-c2cn(CC3CCCC3NC(=O)CCC3CC(C)C3)nn2)cnn1C CCC(C)C(O)C(=O)N1CC(O)(C(F)C(=O)NC(c2c[nH]ccc2=O)C)C1 C1(C(N(C)CC2COCCO2)=O)CCOCCN1C(=O)CN1CCOCC1=O C(=O)(C1Cc2ccccc21)N1CCCC(NC(c2c(C)nc(O)s2)=O)CC1 N1(C(C2C(CC)CCCC2)=O)CCC2(CC2NC(c2cn(C)c(C)n2)=O)C1 CCC(C(=O)N1CCC(O)(CNC(c2ccc(C)c(F)c2)=O)C1)C(C)C c1(N2CCN(C(=O)NCC3CN(CCOC)C(=O)C3)CC2)ccc(C)cc1Cl C1(CCC=C)(C(=O)NCC(C)(C)C)CN(C(C2CCC3CC23)=O)C1 C(=O)C1=NOC2COCC12.N1(c2n(CC)c(CC3CC3)nn2)CCC2COCC2C1 c1(NCc2cn(CC(=O)Nc3ccc(C(=O)O)cc3)nn2)cccc([N+](=O)[O-])c1 N1(C(=O)NC(c2ccc3c(c2)CCO3)C(C)C)CCCc2ccccc21 c1(NC(C2(CNC(C3(OCC)CC3)=O)CCC2)=O)ccc2c(c1)CCC2.OCC C=CC1OCCC1C(=O)N(C)CC1(O)CN(C(=O)CCCNC(=O)OC)C1 C(=O)(C(C)(C)C(C)NC(c1occ2c1CCC2)=O)N1CCC(CCOC)C1 c1(C(N(CCNC(C23CC(C2)C3)=O)CC2CC2)=O)ccc(-c2ccccc2)cn1 CCCC(O)CC(=O)NC1CCCC(NC(c2cccc(C)n2)=O)C1 c1(C(N2CCN(C(c3c(CC)con3)=O)CC2C2CC2)=O)ccc2c(n1)CCC2 c1(NC(C(C)NC(=O)OC)=O)ccccc1S(=O)CC(O)CC C1(NC(C2CCC(=O)NC2)=O)CCC2CC1CN2C(=O)Cc1cc(F)ccc1F C(=O)(CC(C)CC)N1CCC(C(=O)NC(CCC)C2CC2)C1 C12CCC13CCN(CC3)C(=O)CN2C.N1(C(COC)C)CCCC1 c1(C(=O)OCC2CCC(=C)C2)cc2cc(Br)ccc2cn1 C12(NC(C(C(C)(C)C)NC(c3cc(C)oc3)=O)=O)CCC(CC1)C2(C)C c1(C(=O)NC(CN(C(C2(CCC)CCC2)=O)C)C)[nH]c2c(c1C)CCCC2 c1(OC(C)C)cccc(CC(=O)NCCCCCNC(=O)C2=COCC2)c1 N1(CCNC(c2[nH]cc(CC)c2)=O)CCCN(C(C2(C)CC(=O)N(C)C2)=O)CC1 C1(NC(C2CC=C(C)CC2)=O)CN(C(c2ccc([N+](=O)[O-])cn2)=O)CCC1(C)C C=C(C)C1OCCC1C(=O)N(CCC(=O)NCC(O)CCCC)CCO C1(CC(=O)NCC(=O)NCCC(N)=O)CCC2CC12 c1(COC(C)C(=O)N(C2CN(C(c3ccc(CO)o3)=O)C2)C)sccc1Cl C1(CC(=O)N(C2CCCC2)CCN(C(C=C(C)Cl)=O)C(C)C)CC2(CC2)C1 c1(N(C(C#CC(=O)OCC)=O)c2cnn(C3CCNC3)c2)ccccc1F CN1CC(CNC(=O)CC2C=CC(NC(=O)CN3CCC(=O)CC3)C2)CC1=O O=C(CC1C(=O)Nc2ccccc21)NCC(CN1CCCC1)NC(C1SCCS1)=O c1(C(N(C)CC2CCN(C(C(C)C)=O)C2)=O)cccc2cccc(O)c12 N1(C(c2ccc3nccn3n2)=O)CCC2(CCCN(C(c3nc(Cl)cs3)=O)C2)C1 N1(Cc2cccc(C(=O)OCC)c2)CC2(CCN(C(C3CCCN3C=O)=O)C2)C1 C(=O)(CS(=O)(=O)CCO)NC1(NC(C(C)OCC(F)(F)F)=O)CCCC1 c1(-c2c(C)cc(OC(C)C)nc2)c[nH]c2cc(C(=O)NCCc3nccs3)ccc12 N1(C(CC(C)c2ccncc2)=O)CCC(NC(=O)CC2OCCC2(C)C)C(O)C1 c1(C(=O)NC(CNC(C2CC(CC)OCC2)=O)(CC)CC)cn(C)c(C)cc1=O N1(CCS(C)(=O)=O)CC2CCC1C1CN(C(c3cnc4n3CCCC4)=O)CC21 CCCCC(O)C(C)C(=O)NC1(C)CN(C(c2ccc(CC)nc2C)=O)C1 N1(C(CCCOC(C)C)=O)CC2CCCC2C1C(N1CCCOC(C(C)C)C1)=O C1(CCCC)CCC(C(=O)N(C)CC2CCCC(NC(=O)C=CCO)C2)CC1 Cc1[nH]c(C#N)cc1C(=O)NCC1CCCN(C(C2CCOC2C)=O)C1 N1(S(CC(=O)OCC)(=O)=O)Cc2[nH]nc(-c3ccc(C(C)C)cc3F)c2C1 N1(C(c2cc(CC)ncc2)=O)CCN(C(c2coc(O)n2)=O)C(C2CCCC2)C1 N1(C(CCC=CCC=C)=O)CCN(C(c2nnc(C)s2)=O)C(C)CC1C CCCCC(O)C(C)C(=O)N1CC(C(N2CCCC2CC)=O)(CO)C1 c1(CC(N2CCN(C(CC=CCC)=O)C(COC)C2)=O)cccc(S(C)(=O)=O)c1 C1(C(C)C)N(C(=O)C(n2ccc(CN(C)C)n2)C)CC12CC=CC2 C1(C2CC(C(=O)OC(CC(=O)OCC)C3CC3)C2)NC(=O)NC1=O N1(C(CCN(CCC)C)=O)CCN(C(c2ccoc2C)=O)C2(CC2)C1 Cn1nc(C(N2CCC(CO)(NC(=O)CCS(C)(=O)=O)C2)=O)c(Cl)c1Cl C(C(C)(O)CC(=O)NCC1CC2(CC(NC(=O)COCCC(C)C)C2)C1)OC c1(C(=O)NC2CCC(CNC(COCC=C)=O)C2)cccc(SCC(F)F)c1 c1(C(=O)OC)cc(F)c(C)c(S(=O)(=O)N2CCOCC2C(N2CCCC2)=O)c1 n1(CC)cc(C(N2CCCC2CCNC(C23CC(CO2)C3)=O)=O)c2ccccc12 C1(CC=C)(NC(=O)COCC(F)F)CCN(C(C2CC(=O)N(CCOC)C2)=O)C1 N1(C(Cc2cc(C)ns2)=O)CCC(NC(=O)C(C)c2ccco2)C(CO)CC1 CCCCCC(CN(C)C)C(C)NC1CCOC1c1cccc(Br)c1 c1(C(N2CCCC2C(=O)OC(C)(C)C)C(=O)NCCOC)cn(C)nc1C CC1CC(CNC(=O)C2=CCOCC2)CCN1C(=O)CSc1nncn1C C=CC(CCC)CC(=O)N1CC(NC(=O)Cn2cc(CO)nn2)CC2(CC2)C1 C(CC1=CCOCC1)NC(C(Cn1cccn1)NC(c1c(C)sc(O)n1)=O)=O C(=O)(C(C)S(=O)(=O)C(C)C)NC1C2CC(CNC(COC)=O)(C2)OC1 C1(O)(CCNC(CCCN(C)C(c2ccsn2)=O)=O)CCN(C(=O)COC)CC1.C(N)=O c1(C(N2CCC(NC(c3cn(CC)nn3)=O)C2)=O)cccc[n+]1[O-] N1(C(CC(C(=C)C)C)=O)CCC2(CCC2NC(=O)CCc2ncc(F)cn2)CC1 C(=O)(N=c1cc(C2CC2)[nH][nH]1)C1C(NC(c2cccc(C#C)c2)=O)C1 c1(C(N2C(C)C(NC(c3ccc(F)cc3)=O)CCC2)=O)cccc(S(N)(=O)=O)c1 N1(C(C=C(C)C(C)C)=O)CCOC2(CCN(C(=O)C=Cc3cc[nH]c3)CC2)C1 c1(C(N(C2CCOC2)CC)=O)ccc(C(C)C)c(Cl)c1 N1(C(N(C)C)=O)CCN(CCCNC(=O)Nc2cc(C(N)=O)cn2C)CC1 c1(NC(c2ccnn2Cc2cccs2)=O)ccc(Cl)c2c1C(=O)OC2 c1(N2CC3C(C(=O)NC4CCC(F)(F)C4)(C3)C2)ncc2[nH]cc(I)c2n1 C=Cc1cc(C(=O)NCC2CCCCCN2C(=O)Cc2ccc(C)s2)cc(F)c1 n1(CC)ccc(C(=O)NC(C2CN(C(C3CCC(=O)N3C3CC3)=O)C2)C)cc1=O c1(C(=O)NCC2N(C(c3[nH]cc(CC)c3)=O)CCCC2)n[nH]c2ccc(C)cc12 N(C(=NCCC=CBr)NCC(C)(C)C(=O)OC)CCCC(=O)OC S(=O)(=O)(CCCOc1ccc(C(F)(F)F)cc1)NC(C)C(C)(C)c1ccccc1 CCC(C)C(O)C(C)C(=O)N1CCCCC1CNC(=O)C(C)(C#N)CC c1(C(C(=O)NCC2(F)CC(NC(C3(C#N)CC3)=O)C2)O)cccc(Br)c1 C1(C(N2CC(O)(C(=O)OC)C2)=O)CCN(C(=O)CC2CCCC23CC3)C1(C)C N1(C(C(OC)OC)=O)CCCC1(C)CNC(=O)CCCn1cc(C)cn1 Cn1nnc(C(N2CC(NC(=O)CC3CC4(CCC4)C3)C(F)C2)=O)c1C(F)(F)F c1(C(=O)NCC2C(NC(=O)CCC3CC3)COC2)ccc2c(c1)OCC2 Cn1nccc1C(O)C(=O)NCC1COCC1NC(c1cccs1)=O c1(C(=O)NC(CCCNC(CC(=C)C)=O)C)cc(S(N)(=O)=O)c(C)s1 c1(COC)ccc(C(=O)NC2CCCC2NC(=O)CCN(S(C)(=O)=O)C)s1 c1(CCCC(N2CCC(N(CCCC)C)CC2)=O)ccc(F)c(OC)c1 N1(C(COc2ccc(OC)cc2)=O)CCCC(NC(=O)CCCCSC)C(F)C1 c1(C(N(C(C)(C)C)CC(=O)OC(C)(C)C)=O)ccn(C2CC2(F)F)n1 C1(COC)CN(C(=O)C(n2cc(C)cn2)C)CCN1C(c1ccnn1C)=O C=CCCCC(C(=O)N(C)Cc1ccnn1CC)NC(c1cnn2c1CCC2)=O Cn1ccc(=O)c(C(=O)NCC23CCC2CCN3C(=O)Cc2cnc[nH]2)c1 CC(C)(C)C1=NOC(C)(C(=O)NC(c2ccccc2)CNC(=O)C=CC(N)=O)C1 c1(C(N2C(CNC(C(C)CC(N)=O)=O)CC2)=O)nc2ccccc2cc1Cl C1(CNC(Cn2c(C(C)C)nnn2)=O)COCCN(C(=O)CCC(C)(C)N(C)C)C1 C1(C(N(CCC(N)=O)C)=O)COCCN(CC(O)Cc2ccccc2)C1 CCCCCC(O)CC(=O)NCC1CC1C(=O)Nc1cccc(COC)c1C c1(C(=O)NCCC2(C(N(C)CCC3CCCO3)=O)CC2)cccc(C#N)c1 C(CCC(C)(c1nnnn1C(C)CSc1ccccc1Cl)NCC(C)C)OC C1(NC(Cc2cn(C)nn2)=O)CN(C(=O)CC2CC2(C)C)CCC12CCC2 c1(OC(C)C)ccccc1C(=O)NCC(C)NC(c1cc(C2CCOC2)[nH]n1)=O C1(C(N(CCCOCCNC(c2snc(C)c2N)=O)C)=O)CC(=O)NC(=O)N1 c1(C(=O)NC(C)(CNC(c2ccncn2)=O)C2CC2)cc(Br)cc(F)c1F c1(C(=O)NCC(C)NC(c2c(CC)occ2C)=O)cnn2cccc(C)c12 c1(OC)cc(C(=O)N(CCNC(=O)C(C)NC(C)=O)C2CC2)cc2cnn(C)c12 C1(NC(C)=O)COC2(CCN(C(=O)C(C)O)CC2)C1.c1(S)ccccc1 C1(OC)CC2(C1)CC(C(N1CC(N(C)C(C3(F)CCOC3)=O)C1)=O)C2 CN1CCCC1(C)C(=O)NCCCc1cn(C(C)(C)C)nn1 N1(C(=O)NC(N2CCC(OCC)C2)CC)CCC12CC(C)(CC)C2 C1(CNC(c2csc(Cl)c2)=O)CC2(CCN(C(=O)C=Cc3ccccc3)C2)CO1 c1(C(=O)NCCCN(C(C23CC(C)(C2)C3)=O)CC)ccc2c(c1)C(=O)CCC2 C1(C)(CO)CC(F)(F)C1.c1(C(C2C(CC(F)(F)F)C2)NSC(F)F)nnnn1C1CCC1 Nc1nccnc1C(=O)NCC1CCCN1C(=O)C(F)(F)CC1CCCO1 C1(CC(=O)NC2CCC(SC)C2)CC2(C1)CN(C(C1C3CCC(C3)C1C)=O)C2 C1(CNC(=O)Cc2cccnc2)CCCCN1C(=O)C=CC1CC1 c1(C(C(=O)Nc2c(C(=O)NCC)sc(COC)c2)(C)C)cccc(Br)c1C C=CCC(CNC(=O)CCC1CCCN1C(c1cnc(C2CC2)o1)=O)CC(C)C C#Cc1cccc(C(N2CCOC(CNC(=O)C(C)C(C)C)C2)=O)c1Cl C1(C(C(=O)NCCc2c(C)n[nH]c2)C)CCCN(C(=O)CCCn2cccn2)C1 N1(C(CC2C(=O)NC(=N)S2)=O)CCCN(C(=O)C(=Cc2cccnc2)F)CC1 C1(CC)CN(C)CCCN1C(=O)C(C)CN(C)C(C1(C2CC2)CC(=O)C1)=O c1(OCCCC(=O)NCC2N(C(C(C)O)=O)CC3(CC3)C2)ccc2c(c1)CCC2 c1(C(=O)NCCCNC(C23CC(C(C)C)(OC2)C3)=O)ccc(Cl)c(O)c1 C(=O)(CC1=CCCCC1)N(CC(C(=O)NC(C)Cc1cccnc1)C)C c1(C(=O)NC(C2N(C(c3c(C)noc3)=O)CCC2)C)cc(P(C)(C)=O)ccn1 C1(C(=O)NC(CC)C)CC(OC)CN(C(c2cc(C(=O)O)nn2C(C)(C)C)=O)C1 N1(C(CN(C(=O)C(C)(C)C2CCCC2)CCOC)=O)CCc2sccc2C1 C1(CNC(CCC)=O)CC2CCCCC2N1C(=O)COc1ccc(Cl)cc1F C1(CC)(CNC(c2sc(CO)nc2C)=O)CCCN(C(=O)CC(CC)SC)C1 CC1(NC(=O)CCNC(=O)C(F)(F)F)CC(NC(=O)CC2CCOCC2)C1 CC1CCC(C(=O)NC2CC(NC(c3ccn(C4CCCCC4)n3)=O)C2)C1 N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC(C)C(NC(=O)CN2CC3CC3C2)C1 CC1(C)CCCN(C(c2cccs2)=O)C1C(N1CCC2(CC(F)C2)C1)=O C1(C(C)(C)C)(C)CCN(C(=O)CS)C1.c1(C(=O)NC2C(C(C)(F)F)C2)ccoc1 CC(CC(N)=O)C(=O)NCCC(C)(C)NC(C1(Cc2ccccc2F)CC1)=O c1(C(=O)NC(C)C)ccccc1NC(c1cc(-c2cccc(F)c2)on1)=O O=C(C(CC1CCOC1)N(CCCF)CC1CCCCC1)NCC1CCCCC1 O=C1CC(NC(C2CC(CCO)C2)=O)CN1c1cn(CCO)nn1 CC1C(NC(=O)CC2(N3CCCC3)CC2)CCCN1C(=O)Cc1ccnc(F)c1 C(CC1=CCN(C(C2CCNC2=O)=O)CC1)NC(CN(CCC#C)C)=O C(=O)(N=c1cc[nH]c(CO)c1)C12C(CN(C(c3c(OCC)nn(C)c3)=O)C1)C2 N1(C(CCC(=C)Br)=O)CC(C2CN(C(=O)CC(C)(C)F)C2)C1 C1(CC)C(C(=O)NCCn2cnnc2)CCN1C(c1cnn(C)c1CO)=O C(=O)(C(C)CC(=O)NCCCCC1CCN(C(C2CCC(=O)N2C)=O)CC1)OC CCCS(=O)(=O)c1ccc(C(=O)NC2CN(C(c3cn(C4CC4)nn3)=O)C2)cc1 c1(CC)nc2ccccn2c1C(=O)NCCN(C)C(C1(C)CCC(C)C1(C)C)=O n1(CCC(N2CC(NC(CC3N(C(C)C)CCC3)=O)(CO)C2)=O)cccnc1=O c1(CC)nnc2cc(NCC(C3CC3)NC(=O)CC3CCCCO3)ncn12 C1(NC(c2c(CC)n(C)nn2)=O)CC2CC(C1)CN(C(C1CCC(=O)N1C)=O)C2 N1(C(c2[nH]c(=NC)sc2)=O)CCN(C(=O)CCCCCF)C(C)C1C C1(O)(C(C)NC(c2cnc[nH]2)=O)CCN(C(c2c(Br)noc2C2CC2)=O)C1 Cc1cc2sc(C(=O)NCC3CCCN3C(C3CC34CCCCCC4)=O)cc2s1 CC1(NC(c2ccc(CO)s2)=O)CC(NC(=O)CCC2CC2(F)F)C1 C=CCC(CC)C(=O)NCCCCCCNC(C1CC1c1c(C)cccc1C)=O C1(C(=O)NC2CCC(NC(C(CC)(C)O)=O)CC2)CCc2c(cnn2C)C1 c1(C(=O)NC2C(NC(CC(C)F)=O)CCCC2)[nH]cc2c1CCS2(=O)=O c1(C(N2CCC(CN(C)C(C34CC3COC4(C)C)=O)C2)=O)ccnc2ccnn12 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CCCN(C(COCC(=C)C)=O)C(C(C)C)C1 C1(O)(C(C)NC(c2cc(Br)co2)=O)CCN(C(=O)CCN2CCCC2)C1 c1(C(=O)NC2CC(NC(C(CCC)OCC)=O)C2)oc(S(N)(=O)=O)cc1C C1(N(C(Cc2c(OC)nccc2)=O)CC#N)COC2(CCNCC2)C1 C(=O)(CCCC(C)(C)C(=O)OC)N1CCC(CCNC(C(CC)C(F)(F)F)=O)C1 N1(C(CNC(=O)OC)=O)CC2(C)CC1(C(=O)N(C1CC1)Cc1nccn1C)C2 c1(NCc2n(C)cnc2Br)ccc(S(=O)(=O)NCC(C)(C)C(F)F)c(Cl)c1 Cc1cc(C(N2CC(O)(C(C)NC(=O)C(O)CCc3ccccc3)C2)=O)c(C)s1 c1(C(=O)NCCC2(CNC(C3COC3)=O)CC2)cc(N2CCC2)nc(Cl)c1 C1(NC(Cc2c(C(C)C)cccc2)=O)CCC(C)N(C(c2cc(CO)[nH]n2)=O)C1 N1(C(C(CC)F)=O)CC(CO)C2(C1)CN(C(c1ccc(C(F)(F)F)[nH]1)=O)C2 c1(C(=O)NC2(C)CN(C(C3C(CCOC)C3)=O)C2)cccc(C2CC2)c1 C(=O)(CCCCC(C)(C)C)N1CCC(C)C(CC(=O)NCCCCCF)C1 C1(C(=O)NCC2(NC(C(C(C=C)C)C)=O)CCCC2)CC2CCC1CC2OC C1(CNC(C(F)=CC)=O)CC(NC(c2cn(C3CC3)cn2)=O)C12CCC2 c1(C(=O)NCC2(O)CC(NC(CCOC)=O)C2)csc2c(F)cccc12 Cc1ccc(C(=O)C(=O)NC2CC(NC(C3CC3c3ncccc3F)=O)C2)cc1 C(=O)(C1=CCCCCC1)N1CCC(O)(C(C)NC(c2c(C)cc(O)nc2)=O)C1 CC(C)C(F)(CNC(=O)Cc1ccccc1O)C(=O)N1CC2CC1C(F)(F)C2 CS(=O)(=O)c1cc(C(N2CC=CC2Cn2cc(CCCC#N)nn2)=O)co1 C1(CNC(CN(C(=O)OC)C)=O)CN(C(c2ccc[n+]([O-])c2)=O)CC2CCN1C2 C(=O)(C(C(C)(C)C)NC(C1CC1NC(=O)NCc1cccc(Br)c1O)=O)OC C1(C(N(CCCNC(C2C3CCCC23)=O)C)=O)SC2C=CC1CC2 C1(CNC(C=C2CCC(C)C2)=O)CCCCC1NC(C1CC=CC1)=O c1(C(N(CCNC(=O)CC2CCC(OC)CC2)CC)=O)c(C)nn(C)c1Cl C=C(C)CC(=O)N1CC(CNC(c2ccc(CO)s2)=O)(COC)C1 c1(C2CC(NC(C(=O)NC3CCCNC3)=O)C2)ccc(Br)cc1 c1(C(=O)NC(CNC(CN(C)CC2CCCC2)=O)(C)C2CC2)cc2ccsc2s1 C(=O)(C(C(C)(C)O)NC(=O)Cc1cc[nH]c1)NCc1ncc(C)nc1 Cc1noc(C)c1CC(=O)N(CC(C)(C)CNC(c1cccc(CCO)c1)=O)C c1(C(N2CCCC(C(=O)NC3C(CCC)C3)C2)=O)ccc(OC(C)C)cc1F c1(C(=O)NC2(CC=C)CCCN(C(c3cscn3)=O)C2)ccc(C)c(F)c1F c1(C(N2CC(C(C)NC(=O)C(N3CCOCC3)C)C2)=O)cc(Cl)c(F)cc1F C1(C(=O)NC2C(C)CN(C(=O)CN3CCCCS3(=O)=O)C2)CCC2(CCC2)CC1 C1(NC(=O)Cc2ncc(Cl)s2)CCC(NC(C2(Cl)CC2(F)F)=O)CC1 C1(CNC(C(c2ccc(Cl)cc2)NC(=O)OC(C)(C)C)=O)CCCC(N)C1 c1(NCC2C(C)CN(C(C3(F)CCC3)=O)C2)cc(=O)n(C)c(=O)n1C CCCCC(C)(F)C(=O)N1CCC(CNC(=O)CC2CCCOC2)(COC)CC1 C#CCC(C(=O)NC1CC(C)OC1=O)NC(c1ccnn1CCC)=O N1(C(C(C(C)C)O)=O)CC2(COC(CNC(=O)CCCCCN(C)C)C2)C1 CC(CC(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)CC1CC1)CC2)c1ccco1 c1(C(C)=O)cc(C(=O)NCC(O)CN(C(=O)CCc2cncn2C)C)no1 c1(OC)cc(CC(N2CC(NC(c3coc(CO)c3)=O)C(C)C2)=O)ccc1Br C(=O)(CCC(C)(C)F)NC(C(C)C)(C)CNC(C1CCS(=O)(=O)CC1)=O N1(C(c2cccc(N(C)C)c2)=O)CC2CC(NC(c3cnn(C)c3N)=O)CC1C2 N1(C(c2ccc(CC)s2)=O)CCC(C)C(NC(=O)Cn2cc[n+](C)c2)C1 Cc1cncc(C(=O)NC2CC(C(=O)NCCOc3ccc(Cl)cc3)C2)c1 CC1CN2CC(O1)C2=O.c1(C(CF)NC(=O)CN2CCNC2=O)ccccc1 N1(C(CN2CC(C)(OC)C2)=O)CCC12CCCN(C(c1csc(C)c1C)=O)C2 C1(C)(C(N2CCCC(CN(C(Cn3c(C)nnn3)=O)C)C2)=O)CC2CCC(C1)S2 C1(C)(CNC(C2(C)CCN(C)C2)=O)COCCN(C(=O)C2=NOCC2)C1 c1(OC)ccc(C(=O)NCC2CC2NC(C2CC2(C)C)=O)c2ccncc12 N1(C(Cc2c(C)nsc2)=O)CCC(c2cn(CC3CCCN3CCO)nn2)CC1 c1(OC)cc(C)c(C(=O)NC2COCC2CNC(C2CS(=O)(=O)C2)=O)c(C)c1 N1(C(C2(C#N)CC2)=O)CCC2(CCC2NC(c2ccc(Br)o2)=O)CC1 C(C(C)CCO)NC(C(C)NC(C1CCC1)=O)=O.C12(CC1)C(=O)N2 c1(C(=O)NC23COC(CN=c4[nH]nc(CCC)s4)(C2)C3)cc2c(s1)CCCCC2 c1(C(C)C)cc(C(C)(C)NC(=O)CC(C)C)ccn1.C12CC1C(=O)N2 C1(CC(=O)NC2C(C)CN(C(C3(CN(C)C)CC3)=O)C2)Cc2cc(F)ccc2O1 c1(OCCc2cn(C)nc2)cccc(CC2CC3(CC3)C2)c1 Cc1cnnc(C(=O)NCC2(CCNC(=O)CC3SC(=N)NC3=O)CC2)c1 C12(NC(C(CCOC)(C)C)=O)CC(CO)(C1)OC21CCN(C(=O)COC)CC1 C1(O)(CSC)CCN(C(=O)C(C)CC2CCC2)C1.C1(=O)C=CC(=O)N1 C(CN=c1cccc(S(=O)(=O)NC(C(C)(C)CO)C2CC2)[nH]1)(c1cnsc1)N(C)C C1(NC(CC2(CNC(C(C)C3CC3)=O)CC2)=O)CC2CCCCN2C1 c1(CNC(C2C3(CCN(C(=O)OC(C)(C)C)CC3)C2)=O)cnn2c1OCCCC2 C(CCS(N)(=O)=O)(C(=O)O)NC(=O)NC(C(=O)Nc1cccc(C)c1)C CCCC(C(=O)NC1CN(C(c2ncn3c2CCCC3)=O)CC1O)C(C)C N1(CC(=O)NCC(CN(C(C=Cc2n(CC)ccn2)=O)C)O)CCS(=O)(=O)CC1 C(=O)(CCCCCN(C)C(c1cc(NC)ccn1)=O)NC(C=C)C CC(CN=c1[nH]c(=NC(C)CCCO)[nH]c2c1CSC2)c1ccccn1 CC1=C(C)CC(C(=O)NCC2CCC(NC(=O)CN=S(C)(C)=O)CC2)CC1 C1(C(N2CC(O)(CNC(c3cc(CO)[nH]n3)=O)C2)=O)CCCOCC1 C=Cn1nncc1C(N1CCOC(CC(=O)NC(C2CCCCC2)CO)C1)=O c1(NC(C2CC(F)CN(Cc3ccnc(O)c3)C2)=O)cc(Cl)ccc1C(F)(F)F c1(C(N2CC(C(=O)Nc3cncc(C#N)c3)(SC)C2)=O)cccc(C)c1C#N N1(C(=O)NC2CCC(OCCCC)CC2)CC(C)CC(C)C1 c1(C(C(N2CCC(C(CC)NC(c3cc(F)cs3)=O)C2)=O)(F)F)ccccc1C c1(NCCc2c(C)cco2)cc(=NC(C)(C)CC2CCCC2)[nH]c(C(F)(F)F)n1 C(=O)(CCCN=[N+]=[N-])CCn1cc(C2C(C)CCN2C(c2ccccc2F)=O)nn1 c1(C(N2CC(C)(C(=O)NCc3n(C)ccn3)C2)=O)ccc(Br)cc1O c1(C(=O)NCC2CC(F)CN2C(=O)CCN2CCC2)coc(=O)c2ccccc12 c1(NCC(C)NC(C#CC(C)C)=O)ncnc2cnccc12 C(C(C)(C)S(C)(=O)=O)NC(CC1CCC(NC(c2ccc(C(C)=O)[nH]2)=O)C1)=O CN1CC(=O)Nc2ccc(C(N3CCC(C)(C)C3(C)C)=O)cc21 CCC(F)(F)C(=O)NC1CN(C(c2nocc2C)=O)CC1c1ccc(F)cc1 C12(CC(C)(C)C1)C(=O)N2.C(=O)(CCC(C)OC)NC1C(C(=O)OC)OCC1 c1(C(N2CCC(C(N3CCC(=O)NCC3)=O)C2)=O)nccc2cc[nH]c12 C1(CNC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)C2=C(Cl)CC2)CC1 C(CCN(C(=O)Cc1cncnc1)C)(C(C)(C)C)NC(C(CC)OCC)=O C1(=CCNC(c2ncoc2C2CC2)=O)CCN(C(C2CCS2(=O)=O)=O)CC1 C(=O)(C(C)(C)C(C)(C)C)NCC1CCCC(NC(c2c(Cl)cn(C)n2)=O)C1 c1(N(C)Cc2nncs2)ncnc(NC(c2cccc(C)c2)C2CC2)c1C C1(CC(=O)NCC2CCN2C(c2cccc(Br)c2)=O)CC2(CC2)CO1 c1(C(N2CC3CC2CO3)=O)cc2cc(C3=COCCC3)ccc2o1 c1(NC(C(c2cccnc2)C)=O)ccccc1C(=O)N(CCO)Cc1ccccc1 C#CC(C(=O)OC(C)(C)C)(C(F)(F)F)OC.O1NC(=O)OCC1 C(=O)(C(CO)C(F)(F)F)NCC(C)N(C(CCNCC)=O)CC.C(CO)CC c1(CC)ncccc1C(N1CCC(C(=O)NCC(O)(CO)CO)C1C(C)C)=O C(=O)(C(C)C(F)(F)C(F)F)N1C(CN(C(c2ccc(O)cc2F)=O)CC)CCC1 CC(CC(=O)NCC1CN(C(C2CCC(=O)O2)=O)CCC1C)CC(F)(F)F c1(CNC(C(C2CN(C(COC)=O)C2)OC)=O)ccc2ncsc2c1Br C(C)(CNC(c1ncoc1C)=O)(C(C)C)NC(CSCC(=O)OC)=O C1(C(=O)OCC)(COC)CCCN(CC(=O)Nc2cc(CC)ccn2)C1.OCC C12CC3(CC(CCS3=O)NC(=O)OC1)C2.C#CCCCC(=O)OC(C)(C)C c1(CC(=O)NC2C(OC)CN(C(c3csc(C)c3)=O)C2)c(CC)nn(C)c1CC c1(C(C)F)cccc(NC(=O)C(CC2CC2)NC(=O)C2=CCSC2)c1 C1(N(C(COCC)=O)C)CCCCN(C(c2ccc(CC3CC3)cn2)=O)C1 c1(C(N(C2CN(C(c3ccc(C)c(F)c3)=O)CC2O)C)=O)cc2n(n1)CCCO2 N1(C(c2c(C)n(C(C)C(C)C)nc2)=O)CCCC1C1CCCN1C(C1OCCO1)=O c1(C(N2CCN(C(Cc3c(C)n[nH]c3C)=O)CC2)=O)ccc2c(c1)nc(C)n2C C(=O)(C(F)CC(C)(C)NC(C1CCC(=O)C1)=O)N(C)CC1CCCCO1 N1(C(c2c(COC)cc[nH]2)=O)CCC(F)(CNC(C2(NC(N)=O)CC2)=O)CC1 CN1CC(C)(NC(C2CCC=CC2NC(c2cnc(Cl)s2)=O)=O)CCC1=O c1(C(N2CC(N(C(c3c(C)nn(C)c3C)=O)C)C(O)C2)=O)ccnc2cc[nH]c12 N1(C(c2c(C)ocn2)=O)CCCC(NC(C2CCCN2C2CC2)=O)C1C C1(CC(N2C(C)(C)C(NC(c3sccc3CO)=O)CC2)=O)CCCC2(CCC2)O1 C1(C(=O)OC)(N(CCC(C)OC)CC2CC2)CC(c2nc[nH]n2)C1 Cc1c[nH]c2ncc(C(N3CCC(C)(NC(C4CC5C=CC4C5)=O)C3)=O)cc12 C1(NC(C2(SC)CC2)=O)CCN(C(c2cc(-c3ccccc3)cn2C)=O)C1C C(=O)(C(O)C(C)(C)C)NCCn1ccc(C(=O)NCC(C)=O)c1 CCCCC(CC)C(=O)N1CCN(C)C(CNC(=O)C(CCC)OCC)C1 C1(C(=O)NCC2(C)N(C(CN3CC(C)(C)C3)=O)CCC2)CCCCCCC1 C1(NC(C(C)OCC=C)=O)(CF)CCN(C(=O)C=CC(c2ccccc2)=O)C1 c1(NC(C2C=CC(NCc3ccc(F)nc3F)C2)=O)cnc(Cl)c(Cl)c1 C1(NC(C2C(C(C)C)CCC2)=O)CC2CCCC(C1)N2C(=O)C(F)(F)C1CC1 C1(NC(C2(CC=C)CCC2)=O)COC2(CCCN(C(c3cn(C)nn3)=O)C2)C1 C(=O)(CCC(N)=O)N1CC(CNC(CCc2cc(C)[nH]n2)=O)(OC)C1 c1(C(=O)NC(C(C)NC(CCOC(C)C)=O)C)cccn2[nH]c(=N)nc12 C1(O)(C(C)NC(=O)CN(C2CCSC2)C)CCN(C(c2cc(Cl)ns2)=O)C1 c1(OCC(=C)C)ccc(F)cc1.c12nnnn1CCNC2CCC1CCCC1 N1(CC2CCN(C(C(C)CC(=O)c3ccccc3)=O)C2)CCCOC(C)(C)C1 c1(C(=O)NC(C(C)NC(=O)C=CC=C(Cl)Cl)(C)C)ccnc2ccnn12 c1(C(N2C(CNC(C(COC)C)=O)CC3(CC3)C2)=O)cc(=O)n2nccc2[nH]1 N1(C(C)(C)C)CC(C(=O)NC2CCN(CC(=O)Nc3nccs3)C2)CC1=O C(=O)(CCCCC(C)(C)OC)N1CCN(C(C(CN(CC)CC)F)=O)C(CO)C1 N1(C(c2ccc(C)n2C)=O)CCOC2CCN(C(=O)CCOC3CCC3)CC12 N1(C(C2(c3ccccc3Cl)C(C)C2)=O)C2CCC1(CNC(c1ccncn1)=O)CC2 Cc1c(C(=O)NC2COCCC2NC(=O)CC2CCOC2(C)C)sc2cncn12 C#Cc1ccc(C(=O)NC(C)CC(C)NC(=O)COCCc2cccnc2)cn1 c1(NC(C(CNC(c2cnns2)=O)N(C)C)=O)cnc(O)c(F)c1 C(N=c1cc(NCC2CC23CCOC3)nc(C(F)(F)F)[nH]1)c1cnc(N(C)C)s1 C12(C(=O)NC3CCC(CCC)CC3)CCC(CC1)N(C(=O)Cc1ccsn1)C2 C1(OC)CN(C(=O)Cc2cc(C(C)C)nn2C)CC1NC(C1CC=C(C)CC1)=O n1(C(C)C(=O)N(CC(C)(C)C)Cc2cccs2)cc(C2(O)CC2)nn1 N=c1cc[nH]cc1C(=O)NCc1cc(OCc2ccccc2)ncn1 Cc1cc(C(N2CCOC(CCNC(=O)CCCc3cc[nH]n3)C2)=O)ncc1F N1(C(C2C(CNC(C3(CC#C)CC3)=O)C2(C)C)=O)CCn2ncc(O)c2C1 C(=O)(C=C1SCC(=O)N1)C(CC1ON=C(CC)C1)=O.C1(NCC)CCCCC1 C12(NC(=O)C3=CCC3)CCCC1CN(C(C1(CC3CC3)CCC1)=O)C2 N1(C(C=CS(C)(=O)=O)=O)CCC2(CCN(C(C3CCc4nnnn4CC3)=O)C2)C1 N1(C(C2C(C(C)NC(=O)C3=CCSC3)C2)=O)CC2(C1)CC1(CCC1)C2 C1(NC(=O)C=C2CCCOC2)CC2(CCN(C(=O)CC=C(Cl)Cl)C2)C1 c1(C(N(CC(O)CNC(c2ccc(C#N)c(Cl)c2)=O)C)=O)cnn2ncccc12 C1(C(=O)NCc2ccccc2I)CC2CCCCC2N1C(c1cccc(Br)c1)=O C1(NC(C(C)CN=[N+]=[N-])=O)CC2CC(C1)CN(C(C1CC(CC3CC3)C1)=O)C2 CCCS(=O)(=O)C(C)C(=O)NC1CC1NC(c1n[nH]cc1OC)=O c1(SCC(=O)NCCCCNC(=O)CC23COC(CF)(C2)C3)ccc(Cl)cc1 c1(OC)cccc(C(C)CC(=O)N2CCC2CNC(c2onc(C)c2C)=O)c1 C1(CNC(CCc2cnc(C)s2)=O)CCC(NC(C2CN(C(C)C)C2)=O)CC1 C=CC1COCC1NC(=O)CCN(C(=O)Cn1ccc(C)cc1=O)C(C)C C1(C(N(CC(C)NC(C2CC2(C)C)=O)CC)=O)CC2CC(C1)C(C)C2 c1(N2CCN(c3ccc(C#N)cc3)C(CC#N)C2)ncnc2ncc(Br)cc12 Cc1sc(C)c2sc(C(=O)NC3CC3NC(c3cc[nH]n3)=O)cc12 c1(C(=O)NCC(CN(C)Cc2snc(C)n2)C)cc2n(n1)CCCC2 c1(NC(C2CCCCC2)C(=O)OC)ccc(C)cc1.C12CCCN1C2 c1(C(N2CC(NC(C(N)=O)=O)C(F)CC2)=O)cccn2c(CO)nnc12 N1(C(C2(C)CCCNC2=O)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC(O)C1 c1(NC(C(CC)(C)CNC(=O)C(O)COC)=O)cc(C)c(C)cc1C c1(C(N2CCCC(C)(C)C2C(N)=O)=O)ccc2c(c1)SCC(=O)N2 N1(C(C(C)SC(C)C)=O)CCC(CNC(=O)CCn2ccnn2)C(F)(F)C1 C1(C(N2CC(O)(C(C(=O)N(CC(C)O)CCOC)F)C2)=O)CCCCNC1=O c1(OCC)cncc(C(=O)NC2CCCC2CNC(C2CCCS2)=O)c1 CC(C)C(O)CC(=O)NC(C1CC(NC(c2cc(O)ccc2Cl)=O)C1)C C(=O)(C(C)(C)C(C)O)NC(CCCNC(c1c(C)csc1)=O)C c1(C(=O)NC(C2N(C(CCCCOC)=O)CCCC2)C)ccc2nsnc2c1 c1(CC(=O)NCC2C(NC(CCC#C)=O)C2)sc(SC(F)F)nc1C c1(C(N2CCCC(NC(=O)C(F)(F)C3CC3)C2)=O)csc2ccc(Cl)cc12 c1(C(C)(C)OC(C)=O)nc(=NC(=O)N2CCc3ncsc3C2)s[nH]1 C(=O)(C1=CCCCO1)N1CC(CNC(c2cc(C)nn2CC(F)(F)F)=O)C(C)C1 n1(CC)cc(C(N2CCC(SC)C2)CNC(c2ccc(COC)o2)=O)cn1 CC1(C)C2CCC1(C)C2C(N1CCN(C(=O)CNC(=O)Cc2cc[nH]c2)CC1)=O CC1CN(C(c2cccnc2Cl)=O)CCN1C(C1(O)CCOCC1)=O N1(CC(=O)NCC#CCNC(C(COC)O)=O)CCN(C2CC2)C1=O C12(CC(=O)NCC(=C3CN(c4ncn(C)c(=O)c4)C3)F)CCCCC1C2(F)F c1(C(N(CC(C)NC(=O)CCOC2CCOC2)C)=O)ccccc1 c1(CC(=O)NCCOC(CNC(C(CC)=CC)=O)(C)C)cccc2[nH]ncc12 CC1CCc2nc(C(=O)NCCCN(C)C(C3CC3CF)=O)ccc2C1 c1(C(=O)NCC2CCN2C(c2ccc(O)cc2O)=O)cnn2c1CC(F)(F)C2 CC(CC(=O)NCC1CC2CCC1O2)C(C)(C)NC(=O)C(F)=CC1CC1 CN1CCC(C)(C(=O)NCC2CCN(C(=O)C=Cc3ccccn3)CC2)CC1 C(C(O)C(=O)N=c1ccn(CCF)[nH]1)NC(c1nn(CC)c(C)c1)=O C1(NC(CCCOCC)=O)CN(C(C2CCC3(CC3)C2)=O)C2(CCCCC2)C1 c1(C(N(C2CCCN(C(C3C(COC)C3)=O)CC2)C)=O)cccn2ccnc12 CC1(C)COCCC1CC(N1CC(O)(CCNC(C23CCC(C)(C2)OC3)=O)C1)=O C1(NC(C(c2nnsc2C)N(C(C)COC)CC)=O)CCOCC1 C1(c2nc(C)on2)CCN(C(c2ccc(-c3ccccc3)cc2)C)CC1 C1(C(N(CCCNC(=O)C(c2ccccc2)O)CC)=O)CC2CCCN2C(=O)N1 N1(Cc2nc(NC(C34COCCN3C(=O)OC4)=O)sc2)CC2CC(O)CC(C2)C1 c1(NCC2(OC)CCC2)cc(S(=O)(=O)NCC2CC23CCCCC3)ccc1C#N C(=O)(CS(=O)(=O)C1CCCC1)NC1CCC(CNC(C2(C(C)C)CCC2)=O)C1 O=C(CC(C(F)F)n1cccn1)NC1C=CCN(C(c2cnn(CCO)c2)=O)C1 c1(C(=O)NC2CCCC2CNC(c2cc3ccncc3[nH]2)=O)cnc2n1CCCC2 C(C(=O)NC1CCCC1NC(c1sc2nccn2c1)=O)(C(C)O)NC(COC)=O C1(F)(CNC(C2C(CC)C2)=O)CCCN(C(=O)CC(C)F)C1 CC1(F)CCN(C(=O)C(=O)NC2CC23CCCC3)C1 c1(C(N(CCCNC(c2cnncc2O)=O)CC)=O)cc(S(N)(=O)=O)c(C)s1 c1(C(C)(F)F)ccc(C(=O)NCCOCCNC(C2CCCN2C=O)=O)cn1 c1(C)ccc(-n2cc(CN3C(=O)CSC3=S)nn2)cc1.N1(OC)CCOCC1CO C1(NC(CSC)=O)CCC2CCN(C(c3ccc(Cl)nc3)=O)C1C2 C#Cc1cc(C(=O)NCC(C)N(C(c2cn(C)nc2O)=O)CC)cc(Br)c1 CN=c1cc(C(=O)NCC2CC(NC(C3OCCOC3(C)C)=O)C2)cc[nH]1 C#Cc1cc(NC(CC(CC)NC(=O)OC(C)(C)C)C(=O)O)ccc1C c1(SC(c2ccn(CC)n2)=O)ccc(C(N2CC(c3cn(CC)nn3)C2)=O)cc1 C(=O)(C(C)(O)C(C)(C)C)NCC(CNC(Cc1c(C)cc(Cl)cc1)=O)CO Cc1nc(CC(N2CC(C(=O)NCc3cc(C(C)C)no3)C2)=O)n[nH]1 n1(CC(=O)N(CC(C)(C)NC(C(C)C2CC2)=O)C)ncc(O)nc1=O C1(C(N2CC(C)C(NC(=O)CC3CN(C)C3)C2)=O)CCCN(S(N)(=O)=O)C1 c1(C(N(C(C)C(=O)NCCC=CCN(C)C)C2CC2)=O)cn(C)cn1 C(N=c1[nH]c(=N)[nH]c(=NC2CCCN(C)CC2)[nH]1)C1(C)ON=C(C)C1 c1(C(C(=O)NC(C)C)N(CC(COC)C)C)cc2ccsc2n1C C(=O)(C1=CC2(CCN(C(=O)C=Cc3ccoc3)C2)C1)N(C(C)C(N)=O)C c1(C(C(=O)NC2CC2)N(CCCN(C(C)=O)C)C)ccnc(Br)c1 C1(C(=O)NCCCCN(C)C(c2nc(C3CC3)cs2)=O)CCOCC1(C)C C#CCCCCCCCC(=O)N1CC=CC1CNC(=O)CCS(N)(=O)=O CC1=C(C)CC(C)(C(=O)NCC(C2CCCN2C(=O)C2=CSCCO2)(C)C)CC1 c1(C(N2CCC3(CC2)CC3CO)C(=O)NC)cc(O)c(N(C)C)cc1[N+](=O)[O-] N1(C(C=C(C)c2ccco2)=O)CCC2CN(C(=O)C=Cc3ccc(C)o3)CC2C1 CCCCC(O)C(=O)NCc1ccc(-c2ccc(OCC(F)(F)F)cc2)cc1C N1(Cc2cc(C)nn2C)CC(NC(c2cccc(C(F)(F)F)c2Br)=O)C2(CC2)C1 C1(OCC)CCN(C(=O)CNC(=O)CNC(c2cc[n+]([O-])cc2)=O)CC1C CC1CCN(C(C2(n3cnnn3)CC2)=O)CCN1C(=O)C(CO)C(F)(F)F c1(C(=O)NC(CC=C)CNC(c2ccc(C)n2C)=O)cc2cccnn2n1 C1(NC(=O)NCC)CCCN(C(c2cnn(C)c2-c2ccc(OC)cc2)=O)C1 Cc1ccc(CCC(=O)NCCCCN(C(=O)C(O)C2CCCC2)C)c(C)c1 Cc1n[nH]c(C)c1CC(=O)NC1CCCCC1CNC(c1ncoc1Br)=O c1(C(=O)NCC2C(NC(c3c(C)oc(C#N)c3)=O)CCC2)cnc2c(c1)NCC2 C(CCC(C)CC(=O)N1CCC(N(C)C(c2ncn(C)c2C)=O)C1)=C(C)C C1(CC)C(NC(=O)CN(C)C(C)C)CCCN1C(c1cnn(CC)c1)=O C(CCC(=O)NC)NC(CN(CC)CC)=O.C1C(=O)NCCO1 c1(CCC(=O)NC2(C)CC(NC(=O)CC3CC34CC4)C2)ccc(Cl)nc1 c1(C(=O)N)cc(Cl)cc2nc(C)[nH]c12.C1(N(C(=O)CSNCC)CCC)CCCC1 O=S(=O)(CCCF)NC(c1ccsc1)C1CC1 O(NC(=O)C1=CCSC1)CCCC.C(CC(C)CC)NC(=O)C Cc1cnc(C(=O)N(C2CCCN(C(c3ccnc(S)c3)=O)C2)CCO)cn1 C(=O)(C(F)C(C)(F)F)NC(C(=O)NC1(C)CCOC1)CO c1(C(N2CCN(C3CCN(C(COC)=O)CC3)CC2)=O)cnc2sc(C)c(C)n12 c1(N(C2(CO)CNC2)Cc2c([N+](=O)[O-])cn[nH]2)ncnc2ccsc12 C1(C(N(CCCOC)C)=O)CSCN1C(c1ccc(CCCOCC)[nH]1)=O Cc1ccc2c(c1)CN(C(c1ccc3c(c1)OCCO3)C)CC2 c1(N(C(C2CC(C(C)C)OCC2)=O)CCO)ccc([N+](=O)[O-])c(C#N)c1 c1(CN2C(C)(C(=O)Nc3ccc(C)nc3C(C)C)CC2)ccc2sccc2c1 C(N=c1[nH]c2c(F)cccc2o1)C1CN(C(c2cc(OC)nc(OC)c2)=O)C1 c1(C(=O)NC(CCOC)CNC(c2ccsc2)=O)cccc([N+](=O)[O-])c1O c1(N(C)C)ncc(C(=O)NCCC(O)CNC(=O)C(C2CCOCC2)O)o1 CCCCC(C)(F)C(=O)N1CCN(C(c2ccccc2)=O)C(CC(F)F)C1 N1(C(COCCOC)=O)CCCC(CC(N2CCC(OC)C2(C)C)=O)CC1 c1(C(=O)NCC(C2CC2)NC(C(C)n2ccnn2)=O)cccnc1OC(F)(F)F c1(C(=O)OCC)cccc(C(=O)NC2(CNC(c3coc(C)n3)=O)CCC2)n1 CCCC(C)(O)CC(=O)N1CC2(CC(NC(=O)CCC3(O)CCC3)CO2)C1 C1(C2CN(C(=O)COC3CCC(C)CC3)C2)(NC(CCSC)=O)CC1 C#Cc1cnn(C)c1C(=O)NC1CN(C(c2ccccc2CSC)=O)CC1C n1(CCCC(=O)NCCC(C)NC(C2(C)CSC2)=O)c(=O)oc2ccccc12 c1(C(=O)NCCCNC(c2c(N(C)C)ccnc2)=O)cc(O)nc(Cl)c1 S(=O)(=O)(c1ccc(F)c(NC(=O)O)c1)NCC(c1ccnn1C)N(C)C C1(CCNC(CCC(=O)NCC)=O)C(C)CCCN1C(=O)C=C1CCSCC1 CC(=O)CC(C)(C)C(=O)NCC1CCCC1NC(=O)CCc1ncc(C)[nH]1 N1(C(C(CC)CC)=O)C2CCC1CC(CNC(c1cc(C(C)(F)F)ccn1)=O)C2 C1(C(N(C)Cc2cocn2)=O)(NC(=O)CC2COCCO2)CC(O)C1 CCC(CC(=O)NCCN(CC)CC1CC1)OC.C12CC(C1)C(=O)N2C N1(C(C2CCC(C)CC2)=O)CCn2ncc(CNC(=O)C3=CCCO3)c2C1 c1(-c2cc(C)nn2C)ccc2nc(C(N3CCC(N4CCCCC4)C3)=O)sc2c1 Cc1nc(C)c(C(=O)NC2CC(C(=O)NC3CC=CCC3C)C2)o1 Cc1nc(Cl)ccc1CC(=O)NC1(CNC(c2ccc(Cl)nn2)=O)CCC1 CC(C)C(C)(CNC(c1ccccc1CC(C)(C)C)=O)NC(c1ccnn1C)=O C1(OC)CC2N(C1)C2=O.c1(C(C(=O)NC2(CC(=O)OC)CC2)C)ccn(C)c1 Cc1cccc(C(F)(F)C(=O)NC(C)CC2CCN(C(=O)CC3CCOC3)CC2)c1 C1(NC(c2cnco2)=O)CCC2(C1)CN(C(c1sccc1[N+](=O)[O-])=O)C2 C1(CNC(CCNC(C)=O)=O)CCCC1C(=O)N(C)CC1(C)CCC1 C1(N(C(C2CC(C)(C(=O)OC)C2)=O)C)CN(C(=O)CCSC(F)(F)F)CCC1O C1(C(=O)NCCN(C(=O)Cc2ccc(Cl)s2)C)CC2(CSC2)C1 c1(C(N2CCCC(NC(C)=O)CCC2)=O)ccc2c(c1)C=CS2(=O)=O C#CC1CCN(C(=O)CC(C)CNC(c2sc(O)nc2C)=O)CC1 c1(CC(C(=O)OC)NC2CCCC(C)(C)C2)c[nH]c2ccc(F)cc12 C1(C(=O)NCC2OCC(CNC(C(CO)N(C)C)=O)C2)CCC(C2CCC2)CC1 C1(NCCNC(COC(CC)=O)=O)Sc2ccccc2NC1=O.c1(O)cccc(C)c1 Cc1ncn(O)c1C(=O)NC1CC1CNC(C1CC(C(F)(F)F)C1)=O Cn1cnc(CC(O)C(=O)N(C2CCCC2)CCNC2CCC2)c1 C1(NC(C2(C(=O)OC)CC2C)=O)CC2(C1)CN(C(=O)CCc1cccc(F)c1)C2 CC1CN(C(=O)CCc2cc(Cl)cs2)CCCN1C(C12CC1Cc1c[nH]nc12)=O C1(NC(CCN(C(c2ccc(C3CC3)o2)=O)CC)=O)CCOC(C)C1 c1(N2CCC(NC(CC)=O)C2)nc(N2CC3C=CCC(C3)C2)nc2c1ncn2C C1(N=c2nc(NCC(c3cccnc3)(C)C)c3c([nH]2)c(C)nn3C)(CSC)CC1 C(CCCC(F)(F)F)NC(C=CCN(C(c1c(OC)n(C)nc1)=O)C)=O Cc1cncc(C(=O)NC2(C)CN(C(=O)CCCc3n[nH]c(=N)s3)C2)c1C c1(C(=O)NCC(CC=C)NC(=O)CCSCC2CCCO2)cccc(C(C)C)c1 c1(C(N2CC(C)(NC(c3nnn4c3COCC4)=O)C2)=O)ccc([N+](=O)[O-])cc1O c1(CC(c2nccn2C)N(C(=O)NCCCN2CCCC2=O)CC)ccc(F)cc1C Cc1n[nH]c(C)c1C(C)NS(=O)(=O)CC1(C(F)(F)F)CC(O)C1 N1(C(COCCCC)=O)CCCN(C(=O)Cc2cn3ccccc3n2)C(C)C1 N1(C(C2CCC(C)S2)=O)CCC(O)(CNC(C2(C)CC2)=O)CC1 N#Cc1ccc2c(c1)CCCC2C(=O)NC12CCC(C1)N(C(=O)C=CC1CC1)C2 N1(CC(=O)N(C2CC(NC(C(c3c(C)noc3C)CC)=O)C2)C)CCCCC1=O c1(C(N2C(C)CC(O)C2)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 N1(Cc2ccc(C(=O)NC(COC)C)cc2)CCC2CCCC12 C1(NC(CCC(=C)C)=O)CN(c2nc(Cl)ncc2Br)CC2(CC2)C1 CCCS(=O)(=O)CC(=O)N1CCC(NC(c2n[nH]c3c2COC3)=O)C1 c1(C(=O)NCC(CC)NC(c2ccc(CC)o2)=O)cc2c(cn1)OCCO2 C1(CNC(CC(=O)OCC)=O)CC2CCC1N(C(=O)C1=C(Cl)CCCC1)C2 C1(C(=O)Nc2cnc(CCC)nc2)CC2(CC2)CN1C(=O)CCCc1ccccc1 C1(NC(C=CSC)=O)CCN(C(c2nnn(C(C)C)c2C)=O)CC1C c1(CC(=O)N(C2CN(CCOc3ccccc3)CC2O)C)ccc(Cl)cc1I CC1=NC(F)(CNC(=O)CNC(=O)CNC(=O)C(c2cccnc2)O)C=C1 CCC(O)C(C)C(=O)N1CCN(C(=O)C=Cc2ccco2)CC1 C(c1cccnc1)=C(C)C(N1CCC(O)(CNC(c2cnc(N(C)C)o2)=O)C1)=O C1(C(N2CCCC2c2cncc(F)c2)=O)CCc2c(nnn2-c2ccccc2)C1 N1(C(C2C(C)OCC2)=O)CCC2(CCCN(C(c3nnn4ccccc34)=O)C2)C1 N1(C(C(COC)O)=O)CC(C2(NC(C3C(C)C3(F)F)=O)CC2)C1 C(=O)(C(C)C(=O)N1CCC(F)(C(=O)NCc2cc(C)c(C)s2)C1)OC c1(OC)cc(SC)ccc1C(=O)NC1C2CC1N(C(c1cocc1C)=O)C2C N1(C(CCN2CCN(CC)CC2)=O)CC(NC(c2cccs2)=O)CC(O)C1 C(=O)(C=C1SCC(=O)N1CCCNC(=O)CC(C)(F)F)NCCCC(C)N(C)C C1(CNC(C2(CCCC)CCC2)=O)CC(O)CN1C(c1cn(C)nc1O)=O c1(COC)cc(C(=O)NC(C2CCCN2C(=O)COCC(=O)OC)C)n(C)c1 c1(-c2n(C(C=C)C)nc(CC(C)CC)n2)ccc(S(=N)(=O)C2CC2)cc1 C(C(C)(O)CC(=O)N1CC(NC(=O)CCS(C)=O)CC1C)OC N1(C(C)=O)CCc2ccccc2C1CC(=O)N(C)CCNC(=O)C(C)(F)F N1(C(C(c2cccnc2)C)=O)CCC(C2(NC(c3ccc(Cl)cc3F)=O)CC2)C1 C1(C(=O)OC)CC(=O)NN(C(=O)c2cc3cnc(Cl)cc3s2)C1 C1(C(=O)NC2CN(C(c3cnoc3-c3cccs3)=O)CC2F)CCCNS1(=O)=O c1(C(=O)NCC2C(NC(c3cnccn3)=O)C2)cc(C(F)F)ncn1 N1(C(C(CC)C)=O)CC2CN(C(=O)C(C)Sc3ccccn3)CC12 O=C1CCCC(CC(=O)NC23CC(C(N4CC(C(=O)NCC(F)F)C4)=O)(C2)C3)C1 C1(NC(C(=O)OCC)C2CC2)CCC(C(=O)NCc2ccccc2)CC1 c1(OC)cc(=O)n(C)cc1C(N1CC(NC(C2(C3CC3)CCC2)=O)CC(O)C1)=O C1(COC)(CNC(=O)C(F)C2CCC2)CCCN1C(=O)Cn1ncn(C)c1=O C(=O)(CCCC(=O)NCC(O)CNC(=O)C(C)CF)NCCC c1(C(=O)NCC(C(C)C)NC(C(CC)(C)OC)=O)c(F)cccc1F C(C(C)(C)C(F)(F)F)NC(CCC1CC(NC(c2c(CCC)n[nH]c2)=O)C1)=O c1(C(N2C(CNC(C(F)OC)=O)CC2)=O)cc2c(s1)CCCCCC2 CC1CC(N=c2nc(N(C)Cc3cscc3Br)c3cc(Cl)ccc3[nH]2)CS1 c1(C(=O)NCC2CC(CNC(C3CCNC(=O)C3)=O)C2)ccc(C(F)F)nc1 CCC(F)(F)C(C)(C)NC(N1CC2CC(SC)C2C1)=O.C(C)(C)(C)S C(=O)(C1CNC(=O)c2ccccc21)NCC1(C(C)NC(c2cnccn2)=O)CC1 N1(C(c2c(C)[nH]cc2)=O)CCCC(n2cc(C3CC34CC4)nn2)C1 N1(C(CSCC)=O)CC(F)CC1CC(=O)NCC1CCN(CCF)C1 C1(C(N(C2CCCN(C(C3(Cl)CC3)=O)C2)C)=O)CC(C)(C)CN1C C1(C(=O)NCCCC2N(C(c3scc(C(N)=O)c3)=O)CCC2)C2CCCCC12 N1(C(c2c(Cl)cn(C)n2)=O)CCC(C2(NC(=O)C=CCOCC(F)(F)F)CC2)C1 CCC(COC)(CC)C(=O)NCC1CCCC1C(=O)N(CC(O)C1CCC1)C CC(C(C)(C)C(=O)N1CCC(CC(F)F)C1)NC(c1nn(C)cc1Cl)=O N1(C(C2CN(C(C(CCCCC)F)=O)CC2C(C)C)=O)CCc2ccncc2C1 n1(CC)cc(C(=O)C(=O)NCC(C)(CO)NC(C2CC2C#N)=O)cn1 C1(C(=O)NC2(CNC(CCC#CC)=O)CCCC2)CC(=O)c2ccccc2C1 C(c1ccc(Cl)nc1)=CC(N1CCN(C(=O)C2=CCCO2)C(C(=O)C2CC2)C1)=O C1(NC(=O)Cc2nnc(O)s2)CN(C(C23CC(F)(C2)C3)=O)CC12CC2 c1(N2CCN(C(CC)C)CC2)ncc(C)cc1S(=O)(=O)NC1CC(C)(C)C1 n1(CC(=O)NCCC(C)NC(C2CC3(COC(=O)N3)C2)=O)cc2ncccc2n1 C(CCCCC(=O)NCCC(c1cnccn1)CC)N(N1CC2(CCC2O)C1)C=O c1(C(N2CC(C(C)NC(=O)C=CC3CCCO3)C2)=O)cc(Cl)c(Cl)c([N+](=O)[O-])c1 C(=O)(C(CO)C(F)(F)F)NCC(CCOC)NC(c1cccc2[nH]ncc12)=O c1(CNC(CCOCC#C)=O)cc2n(n1)CCN(C(=O)Cc1scnc1C)C2 c1(C(=O)NCC2CCCN(c3nccc(CC)n3)C2)[nH]c(=O)cnc1C Cc1ccc(CC(N2CC(CF)(NC(=O)C(C)c3ccsc3)C2)=O)c(Cl)c1 c1(OC)ccnc(C(N2CCC(O)(CNC(C3CCN3C(C)=O)=O)C2)=O)c1O C(=O)(C(C)(C)C(=O)NCC1CCC(NC(=O)Cc2ccc(F)c(C)c2)C1)OCC N1(C(N2CCC(OC)C(C)(C)C2)=O)CCN(C)c2cc(F)ccc21 Cc1ccc(CC(=O)N(CCCNC(=O)CN(C)S(N)(=O)=O)CC2CCCC2)cn1 c1(C(=O)NC2CCC(NC(C(C)(CO)OC)=O)C2)cc2sc(C)cc2s1 c1(C(c2n(CC)nnn2)NCc2cn(C)nn2)cccc2c1CCC2 c1(COC)nc(C)cc(=NC(C)CCNC(c2c(C)cccc2Cl)=O)[nH]1 c1(NC(C(=O)NC(C(=O)NC)C)C)ccc(-c2nnnn2-c2ccccc2)cc1 CCC(CC(=O)NC1CC(F)CN(C(c2ccnn2CCOC)=O)C1)C(C)(C)C c1(N2CC(C(C)NC(c3ccc(OC)cc3)=O)OCC2)cncc(C#N)n1 C(C)(C)(CCCNC(=O)CC1CCC(=O)N1C)NC(CCOCCOC)=O C1(C(=O)OC)CC2(CCOCC2)CN1C(C1CCC12CCCO2)=O CC1=C(C(=O)N(C)CC=CC(N2CC(C)CC2CO)=O)CC1 c1(N(C)C(C2CCN(C(=O)C(F)(F)Cl)C2)=O)cc(C(F)(F)F)nn1C N1(C(COC(CCC)C)=O)CC2CCC(C1CO)N2C(C1CCCN1CC)=O N1(C(c2occ(C(N)=O)c2)=O)CCC2CCC12CNC(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NCC2(F)CCCN(C(C(C=C)(C)CC)=O)C2)cc2sc(C)cc2[nH]1 Nc1ccc(Cl)c(C(=O)NC2CCCCC2NC(C23CCC(CC2)C3)=O)c1 c1(C(N2C(CNC(C(F)=CCC)=O)C=CC2)=O)cc(O)cc([N+](=O)[O-])c1 C1(C(=O)NC2(C)CCCN(C(c3ncc(Cl)cc3Cl)=O)C2)CCOC2(CCC2)C1 C12(C(N3CCC(NC(CCC4OCC(C)(C)C4)=O)C3)=O)CC3CC1C2C3(F)F C1CCC(=O)N1.c1(C(=O)OC)nc(C(=O)N(CCO)CC2(O)CC2)cs1 Cc1ncc(F)c(NC(C2CC3(C2)CN(C(=O)C(O)CC(C)C)C3)=O)n1 C(=O)(CCC(=O)N1CCCC1CN(C(=O)C(Cc1ccccc1)SC)CC)OCC C1(CNC(c2cc(OC)cc(F)c2)=O)CC2(CCN(C(=O)C3=CCC3)CC2)CO1 C(C1=CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)CC1)NC(c1cc(Cl)cs1)=O c1(-c2nc(CC(=O)OCC)c(C)s2)cc(OC)ccc1OCOC N1(C(C(C)=CC)=O)CC(NC(=O)C(C(C)C)n2cc(C)cn2)C(C(F)F)C1 N1(CC(=O)NCc2cn(-c3ccc(OC)cn3)nn2)CCOc2ccccc21 C(=O)(C#CC1CCOCC1)N1CC(NC(=O)C(C)Cc2cnc[nH]2)CC(C)C1 Cc1cccc(C(N2CCCC2(C)C(=O)NCCc2ccc(O)c(O)c2)=O)c1I Cc1onc(C2CC2)c1C(=O)OCCc1csc(NCC2CCCN(C)C2)n1 N1(C(CC(C(C)OC)NC(=O)CC2(O)CCOC2)=O)CCC2(CCC2)CC1 CC1CC(N=c2ccc3nnnn3[nH]2)CN1C(=O)CCCCCS(N)(=O)=O Cc1ccn(CC(=O)NC2COCC2CNC(=O)C(C)(C)C(N)=O)c(=O)c1 C(N=c1nc2sccc2c(N2CCc3c(cnn(C)c3=O)C2)[nH]1)c1nc(C)sc1 C1(NC(c2c(CC)c[nH]c2)=O)CC12CCN(C(C1COCCN1C)=O)CC2 C1(C(=O)NCCCC(C)C)CCCN(C(c2ccccc2N2CCCC2)=O)CC1 c1(CN=C(NCC(CC)OC)NC2CCCCC2)ccc(O)c(Cl)c1 C1(NC(C2CN(C(C(C(C)(F)F)F)=O)C(C)(C)C2)=O)CCCOC12CCC2 CC(C(=O)NCC1CC1NC(=O)CN(C)Cc1cocn1)n1ccnc1 Cc1ccc(NC(C2CCOC2CNC(C2Cc3nccn3C2)=O)=O)c(C)n1 c1(SSCCNC(=O)NCC2CCCC2)ccnc(Br)c1 C=C(C)CC(C(=O)NC1CCCN(C(c2scc(Cl)c2Cl)=O)C1)NC(C)=O c1(COC)noc(C(=O)NCC(C2CC2)N(C(=O)CC(=O)NC2CC2)C)n1 C(=O)(CC1OCCc2ccsc21)NCCN(C(c1c(CC)occ1)=O)CC c1(C(=O)NCC(F)CNC(C2CC3CC3C2)=O)cnc2ccccc2c1 c1(CC)ccc(C=CC(=O)NC2CC(NC(C34CC(C)C3C4)=O)C2)o1 c1(OCC(=O)NCC(n2cc(CC=C)nn2)C)ccccc1C C#CC1(C)CCCN(C(C2C(O)CCN2C(c2cc(C(C)C)[nH]n2)=O)=O)C1 C1(NC(C2CCN(C(c3c(O)cccc3F)=O)CC2)=O)CCn2cnnc2C1 C1(NC(CCc2cc(C)no2)=O)CS(=O)(=O)CC1NC(c1ccc[nH]1)=O N1(C(CC2CC(OC)C2)=O)CCCCC(N(C)C(c2cnn(C(C)C)n2)=O)C1 C1(C(=O)NC2CN(C(CCSC)=O)CC2C)CCc2ccc(F)cc2O1 CC1(C)C(C)(C)C1(F)C(N1CCC(CO)(NC(=O)CCN2CCCS2(=O)=O)C1)=O Cn1c(=O)ccn(CC(N2CCCC(CS(C)(=O)=O)C2)=O)c1=O N1(C(C(C)(C)CF)=O)C2CCC1C(CNC(C1(C)CC1Br)=O)C2 C1(CC)CCCN(Cc2cccc(C#N)c2)C1C Cc1ccc2occ(C(=O)NC3CCN(Cc4cnn(C)c4Cl)CC3(C)C)c2c1 CC1COC(C)(C(=O)NC2CC2NC(=O)CCNC(=O)CO)CO1 c1(C(=O)NCC2C(NC(C3(C)CC3)=O)CCC2)nc(C#N)cs1 N(C1CCCc2ccc(C(C)C)cc21)S(c1c(OC)ccc(Cl)c1)(=O)=O C(=O)(CCC(F)(F)C(F)(F)F)N1CC(CCNC(c2c(CC)nc[nH]2)=O)OCC1 c1(SCCC(=O)NCCC(C)NC(C2(CF)CCOCC2)=O)ccc(Cl)cc1 c1(Sc2ccccc2)cccc(-n2cc(C(C)N(C)C(C3C(C)C3)=O)nn2)c1 Cc1ccc(CNC(=O)C(C)N(C(=O)CCc2cncn2C)C2CC2)nc1C C=CCCC(C(=O)OC)NC(=O)C(CCC)NC(=O)CC1COCCO1 C(=O)(C1=CC2(CN(C(=O)C(C)(C)CCCF)C2)OC1)NC(CC)(C)CO c1(C2(OC)CCC2)nc(NC(c2cnc(-c3ccccn3)nc2)=O)cc(O)n1 C1(CN(C(=O)CCN2CCC(F)C2)C)CCN(C(c2scnc2Cl)=O)C1 c1(C(N(CCNC(C(c2ccc(C)cc2)C)=O)C)=O)cccc2cnnc(O)c12 N1(C(CCC=C(C)C)=O)CCC(C(CO)NC(=O)C(C)(C)CN(C)C(C)C)CC1 N1(C(c2c(C)ncs2)=O)CCC2(CC1)CC2CNC(C1(F)CC1(Cl)Cl)=O C(=O)(C1CCCc2ccnn21)N1CC(Nc2ncc(O)cn2)CC(C)C1 N12CCC(S(=O)(=O)NC(CCC)C1=O)C2.C1(C(=O)OC)CC1 C(=O)(C1SCc2cccnc21)NCC1(OC)CN(C(=O)CN2CCC(C)(O)C2)C1 CP(C)(=O)c1ccc(C(N2CCOCC2CCNC(C2CC(CC3CC3)C2)=O)=O)o1 CN1CCCC1C1COCCN1c1cc(Cl)ccc1S(N)(=O)=O N1(C(c2n(C)cnc2)=O)CCC2(CC2C(N2CCCN(CCO)CC2)=O)C1 c1(NC23CCC(C(=O)OCC)(CC2)C(C(=O)OC)O3)c(C)[nH]c2c(OC)cccc12 Cc1cc(C(=O)NCC23CCC(NC(=O)CSC(C)(C)C)(CO2)C3)cc(F)c1 C1(C)(NCc2n(CC(=C)C)nnn2)C(C)(C)C1(C)C n12cc(c(=O)cc1C)NC(=O)C2.C(CCC(C)NC(C1(N(C)C)CC1)=O)SC C=CC1CCCC(NCc2noc(-c3cccc(C)c3)n2)C1 C1(CNC(c2cc(C)nn2C)=O)CC2CCC1N(C(=O)C(C)NCC(F)(F)F)C2 C1(NC(c2cnn(C3CCCC3)c2)=O)CCC12CCN(C(=O)C=C1CCC1)CC2 Cc1nocc1CC(N1CCCC1C(C)NC(C1(n2cncn2)CC1)=O)=O c1(N(CCC(C(F)(F)F)OC(F)(F)F)C=O)cnc2c(Cl)cnn2c1 c1(C(=O)NC2C(C(N3C(CC(=O)OC)CCC3)=O)CCC2)cc(CO)ccn1 N1(C(=O)Cn2cc(C3OCCO3)nn2)CCC(Cc2ccccc2)C(F)(F)C1 CC1(C(N2CCC(C(O)CNC(c3cc(Cl)ns3)=O)CC2)=O)CCCOC1 C1(C(=O)NC(C2CCN(C(c3cn(C)nn3)=O)CC2)C)CCc2nnn(C)c2C1 C1(NC(c2cc(C3CC3)no2)=O)CC2CCC(C1)N2C(=O)CCCc1cncs1 N1(C(C2CCCC2)=O)CC2(CCN2C(C2CCCS2)=O)C1 Cc1ccc(F)c(CN2CC(C(=O)NC3CC(O)C3)CC(F)C2)c1F CN(CCCC(=O)N1CCN(C(C2CCCC2C2CC2)=O)CC1)N=O.C1C(=O)N1 N1(CC(=O)NCCC(=O)NC)CCc2cc(OC)cc(C(F)(F)F)c21 Cn1nc(C(N2CCCCC2CNC(=O)CCc2cnco2)=O)c(Br)n1 C1(OC)(CO)CCSCC1.c12ncc(s1)CC(=O)N(C)CCCNC(=O)NCC2 C(CC(=O)NC(C1(Nc2ncc[nH]2)CC1)C)N(C)CC.C1C(=O)NCCO1 C1(CNc2ccc(C(c3ccc(F)cc3)O)cc2)CN2CCCC2CO1 C(CCCCCC(=O)NCC1CCOC(C)C1)NC(C(CC=CCC)C)=O C=CC(C)(C)CC(=O)NC1CN(C(=O)Cn2cc(C3CCOC3)cn2)CC1F C=C(Br)CC(=O)N1CC(COC)(NC(=O)C(Cl)=CCl)C1 CCCC(C)CCCC(=O)N1CCC2(CCCN2C(=O)COC2CC=CC2)C1 N1(C(CC=C=C)=O)CCC(NC(=O)Cn2cc(C3CC3)nn2)C(O)C1 S(=O)(=O)(c1cccc(C(N2CCC3(CC3)C2)=O)c1)Nc1ncc(C)nc1 c1(OC)ccc(Br)cc1CN(C(C1COC(C)(C)O1)C(=O)NCC1CC1)C1CC1 n1(CC(N)=O)cc(C(=O)NCC2C=CC(NC(c3ccnn3C(F)F)=O)C2)nn1 Cn1ccc(C(N2CCCCC2C2CCN(C(c3csc(Cl)c3)=O)C2)=O)cc1=O C1(NC(c2ccc(OC)nc2)=O)CC2CC1CC2N(C)C C12(CNC(c3c(COC)ncs3)=O)CCC(C1)N(C(C1(C)CC3(CCC3)C1)=O)C2 Cc1cccc2[nH]cc(CCC(N3CCC(C(C)NC(=O)CC4CSC4)C3)=O)c12 N1(C(C(=Cc2ccccn2)C)=O)CC2CC(NC(=O)C=Cc3ccco3)CC1C2 C1(CNC(c2cc(C#C)no2)=O)COC(C(F)(F)F)CN1C(=O)C(C)(F)F N1(C(C2CC(C(N)=O)C2)=O)CC(NC(c2ccnc(C3CC3)c2)=O)CC2(CCC2)C1 c1(CN(C(C(C(C)C)OC)=O)C)cc(C)cc(C)c1N.C12CCCC(C1)NC2=O c1(C(=O)NCC(C)N(C(c2coc(C#N)c2)=O)CC)cnc2c(c1)c(C)nn2C c1(CCC(=O)NC(CC(C)NC(CC(=C)Br)=O)C)ccc(OCC)cc1 N1(C(c2[nH]cc(C)c(=O)c2)=O)CC2CCC1C(CNC(=O)CC1CCOC1)C2 c1(SC)cn(C)nc1C(=O)NC1CC(CNC(C2CCOC2C)=O)C(O)C1 C1(C(=O)NCC2CC(NC(C3N(CC)CCCC3)=O)C2)CC2(CCCC2)C1 c1(OCC)ccc(C(=O)NC(C)CCNc2snc(Cl)c2C#N)cc1C c1(NC(c2ncc[nH]2)CC)nc(N(C)Cc2cc(Br)ccc2F)c2sccc2n1 C1(CCC=C)(C(N2CC3CC3C2)=O)CN(C(=O)COCC(=C)C)C1 C1(C(N2CCC(C)(NC(CN(S(C)(=O)=O)C)=O)C2)=O)CCc2nnnn2C1 C=CCCC(C(=O)NCCn1cnnc1CC)NC(=O)C(C)NC(=O)NC C(C1c2ccsc2CCN1C(=O)CCCS(N)(=O)=O)NC(CNS(C)(=O)=O)=O C1(NC(CSC)=O)CCCC(N(C)C(c2nnn(-c3ccccc3)n2)=O)C1 CCC(CC)(C(=O)NC1CCCC1CNC(=O)C(O)C(C)(C)C)OC N1(C(C(CC)N(C)C(c2ccc(C3CC3)cn2)=O)=O)CCC(OC)CC1 c1(C(=O)NC(CC)CN(C(=O)Cc2ccsc2C)C)cc(F)c(F)cc1N c1(CCC(=O)NC(CNC(C(CO)OC)=O)C2CCC2)cc(C)cc(C)c1 c1(C(=O)OC)cc(=NCC2CCCC2NC(c2nc(O)sc2C)=O)[nH]c(Cl)n1 C(=O)(CCCCCS(N)(=O)=O)NCC(C(C)C)NC(c1cnc2n1CCC2)=O C1(CC#C)(C(=O)NC(C)C(C)(C)CN(C)C)CCN(C(c2c[nH]ccc2=O)=O)C1 c1(C2CCN(C(c3c(CC)nc(C)s3)=O)C2)cc(C)n(-c2cccc(F)c2)c1C CC(C)(F)CCC(=O)NCC1(C)CCCN(C(C2(F)CCCC2)=O)C1 C1(NC(CC(=O)NCC#C)=O)CCC(CC(=O)NC2CCCCC2C(C)C)CC1 N1(C(c2cc(CC)on2)=O)CCN(C(=O)CC(O)CN(C)C)CCC1C c1(CC(=O)NCCN(C(C(C)SCC)=O)CC(C)O)ccc2oc(C)nc2c1 N(C1CN(C(c2ncc(OC)cc2F)=O)CCc2ccccc21)C(CCC)=O c1(OC)cccc(C(CNC(c2oncc2C)=O)NC(C23CCC2C3)=O)c1 N1(C(c2cnc(C)[nH]2)=O)CCOC(CCNC(=O)C(CO)NC(=O)C(F)(F)F)C1 c1(CNC(CNC(=O)OCC)=O)oc(CC)nc1C.N12CCC(C)(C1)C2=O CCCCC(F)C(=O)N1CCC(C)(C)C1CC(=O)NCCC1=CCCCC1 C(C(=O)NOCCCC1CC1)(N(C)C(C1CC(C(N)=O)C1)=O)C1CC1 C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C(N(C)C(C2CC2(C)C)=O)C1 c1(CC)cc(C(=O)NC2CC(F)(CNC(=O)CC(C)OC)C2)cc(F)c1 CC(C)(C)C(C(=O)N1CCCCC1CCNC(=O)CCCF)c1ccc(O)cc1 Cc1nccc(C(=O)NC2(C)CC(NC(=O)CCCn3ccccc3=O)C2)c1N N1(C(C2CCC(NC(=O)CNC(c3ccsn3)=O)C2)=O)CCn2ccnc2C1 Cc1cc(N2CCCC(NC(=O)Cc3ncncc3Br)C2)n(C)n1 c1(C(=O)NC2CC(CC(=O)OC)C2)cccc2c1OC(C)C2.C12CCC1NC2=O c1(C(CNC(c2csc(COC)n2)=O)NC(C(CC)C)=O)cc(F)cc(Cl)c1 c1(C(=O)NC2C(CNC(C(N3C(CC)CCC3)=O)=O)C2)cccc2c1OC(C)C2 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)CCCC(=O)OCCC)CC1C(F)F C1(NC(C=CC=CC)=O)CC12CCN(C(c1ccc(C3CC3)nc1Cl)=O)CC2 c1(CN2CCN(C(c3ccc(CC)nc3)=O)C3C2C3)cc([N+](=O)[O-])ccc1Cl C1(OC)CC(CNC(c2n[nH]cc2C)=O)N(C(c2c[nH]nc2C)=O)C1 C(=O)(CC(C)(C)C(F)F)NC(CC(=O)NC1CC(C(C)C)C1)C(C)C S(=O)(=O)(c1cc2oc(=O)[nH]c2cc1F)N1C(C(=O)OCC)CC(C)CC1 N1(C(c2c(OC)nc(C)s2)=O)CC(O)CC1(C)C(=O)NCCCCC(F)(F)F c1(CN=C(NC(COC)C)NC2CC23CCOCC3)cccc2nn(C)cc12 N1(C(C(C)N(c2ccc(Cl)o2)C)=O)CCC(NC(=O)Cn2cnc(=N)[nH]2)CC1 Cc1cc(C(N2CC(NC(=O)C(C)(C)CC3CC3)CC2CO)=O)nc(O)c1 N1(C(CCN2CCC(C)CC2)=O)CCCC(C)(NC(C2CCCCCCC2)=O)C1 C=CC(CCC)CC(=O)N(CCCOCCNC(c1cc(F)c(Cl)cc1Cl)=O)C C1(NC(c2ccon2)=O)CC2CC(NC(C3CCC3c3ccc(F)cc3)=O)C1C2 N1(C(C(C)CC(N)=O)=O)CC2CCC1(CNC(=O)CNC(C1CC1C)=O)CC2 c1(C(N2CC3(C(NC(CC(C)(C)OC)=O)CC3)C2)=O)cc(F)c(F)c(O)c1F C1(OC)C(C(=O)O)CN(C(=O)CN2CCCC2C)C1CSC(C)(C)C C1(CNC(c2n[nH]c(C)c2Cl)=O)CN(C(=O)C(C)(C)N(C)C)CCC1C c1(C(=O)NC(C2OCCN(C(CNC(=O)OC)=O)C2)C)cc(=O)c(OC)c[nH]1 C1(CNC(c2ccc(CO)s2)=O)COCCN1C(c1coc(C2CCCC2)n1)=O C1(SC)CCC(C(N2CCC(N3CCCC3CNC(=O)NC=O)CC2)=O)CC1 C(C(O)CC(=O)N(C)Cc1cccc(F)c1)NC(C1C(C(=O)OC)C1)=O Cc1c(F)ccc(Cl)c1CC(=O)Nc1ccnc(C(=O)OC(C)(C)C)c1Br CCC(=O)CCC(=O)NC(C)(CC)C(=O)NCC(CO)OC c1(C(=O)NC2CC(NC(C(C(=O)NCC)(C)C)=O)C2)cc(O)c(OC)c(C#N)c1 N1(C(CCCOC(C)C)=O)CCC(NC(=O)CCCN(C)C)C12CCCC2 c1(C(C(=O)N(C2CCN(C(C3CC34CCOC4)=O)C2)CC)C)ccc(C#N)cc1 c1(C(=O)NC2C(CNC(c3cc(C)nc(O)n3)=O)C2)ccc2oc(C)nc2c1 C(C(C)(C(=O)NC1CC(C)(O)C1)NC(C1C2CC(=O)CC12)=O)SC c1(OCC=C)ccc([N+](=O)[O-])c(C(N2CC(CNC(=O)C(C)(C)O)C(C)C2)=O)c1 c1(C(N2CCC(O)(CNC(C3(COCC)CC3)=O)C2)=O)ccc2nn[nH]c2c1O c1(OC)ccccc1NC(C1CC(C)CN1C(=O)Cc1ncccc1C)=O N1(C(CC2(C)CN(C(=O)C3=CCSC3)C2)=O)CCOCC1C1CC1 C(=O)(C(F)C(C)CNC(c1ccncc1)=O)N1CCC(CCC#C)CC1 C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(=O)CC(=O)NCC)CC2)C1 c1(C(=O)NCC(CNC(C(C)OCCOC)=O)C)cccc(NC2(CO)CC2)c1 Cc1n[nH]c(C)c1CCC(=O)NC1CCC(NC(=O)C(C)n2ccnc2)CC1 c1(C(=O)NCC2(C)CCC(NC(C(CC)OCC)=O)CC2)cc(C)c(F)cc1F c1(OCC)ccc(CCC(C)NC(c2cnc(-c3ccccc3C)s2)=O)cc1 C1(N(C(=O)C=CC(F)(F)F)CCO)CCN(C(=O)CCCn2ccnc2)C1 c1(OCC(=O)NC2C(NC(C3(C)CC(F)(F)C3)=O)C2)ccc(F)cc1Cl CC1CCC(O)C(NC(c2cn(CCNC(=O)CCNC(N)=O)cn2)=O)C1 N1(C(c2cc(C)ncc2C)=O)CCN(C(C2(F)C(C)(C)C2(C)C)=O)CC(C)(C)C1 CC1(NC(=O)CC2CCCC2)CCCN(C(=O)CCS(C)(=O)=O)C1 C1(C(N2CCC(CC(N3CCC(C)C3CO)=O)CC2)=O)CC2(CCO1)CC2 c1(C(N2CC(O)(C(C)NC(C3C(=C)C3)=O)C2)=O)c(C(=O)OCCOC)cccc1C C1(NC(c2cc(CO)on2)=O)CC2CCC(C1)N2C(C1C=CCS1)=O N1(C(C(CC)(F)F)=O)CC2CN(C(c3cn(C)nc3C(C)C)=O)CC2C1 c1(CC)cc(C(N2CC(CO)(CNC(C3CC4CCC(C3)O4)=O)C2)=O)ccc1F N1(C(c2cc(COC)on2)=O)C2CCC1CN(C(=O)CSc1n[nH]c(C)n1)CC2 C1(NC(C=C(C)C2CC2)=O)CN(C(=O)CCCC(C)C)CC(C)(C)C1 c1(CC)c(C(=O)NCC2C3CN(C(c4cccc(C)c4N)=O)CC23)cccc1F C1(CC(=O)NC2(C3CCCN3C(C3CC=CCO3)=O)CC2)CCCCCCC1 Cc1nc(C)c(C(=O)NCC#CCNC(c2ccc(C(C)(C)C)nc2)=O)o1 C(=O)(CC(O)C(C)(C)C)NCC1(F)CCCN(C(c2nc(C(C)=O)sc2)=O)C1 c1(C(N2CC(CC(CNC(C3C(=C)CC3)=O)(C)C)C2)=O)ccc(SC(F)F)cc1 Cc1[nH]nc2c1CC(C(=O)N(CCO)CCN(C)CCO)CC2.C1(C)C(=O)N1 c1ccc(F)cn1.C1(C(=O)NCSC)(CNC(C=CC(=O)OCC)=O)CCCC1 c1(CNC(N2CCN(c3cccc(OC)c3O)CC2)=O)cc([N+](=O)[O-])ccc1C C(=O)(CC(O)CC(C)(C)C)N(CC(C(=O)Nc1c(C(C)C)nccc1)(C)C)C C1(CN(C(CCOC)=O)C)CCCN(C(=O)CC(C)(C)OCc2ccccc2)C1 Cn1cc(C2=NOC(C(=O)NC3CN4CCC3C4)C2)cn1 C(CCCCCNC(=O)CC1(C)CC1(Cl)Cl)N(C)C(c1cc(CC2CC2)on1)=O C(C(O)(C(=O)NC1CC(NC(c2coc(O)n2)=O)C1)C(F)(F)F)N(C)C C1(CNC(c2ncn(CC)n2)=O)(CO)CCN(C(c2ccnc(O)c2F)=O)CC1 c1(CCC(=O)NC(C(C)NC(CCCSC)=O)(C)C)ccc(Br)cc1 c1(-c2n(CCC=C)nc(CS(C)(=O)=O)n2)cn2ccc(F)cc2n1 C(=O)(C1=CCCCC1)NCC1C(C(=O)Nc2cc(-c3cn(C)nc3)on2)C1(F)F C1(C(=O)NCC2C(NC(C=CC(CC)=CC)=O)CC2)COc2ccc(O)cc2O1 c1(C(N2C(CN(C(C(C)CC(N)=O)=O)C)COCC2)=O)ccn2ccccc12 C#CC1CC2CCC1N(C(C1CCCCC1(C)NC(C1OCCOC1C)=O)=O)C2 c1(OCC(=O)NCC2CC(C)N(C(c3nncs3)=O)C2)cc(Cl)ccc1Cl S(=O)(=O)(c1cccc(F)c1)NCC(=O)NCC1CC2CCC1N(C(=O)C(N)=O)C2 N1(C(c2c(C)noc2C2CC2)=O)CCC(NC(=O)CCC2CCC2)C(F)C1 C1(CC=C)(C(=O)OC)CCN(C(=O)NCC(c2nccn2C)CC)C1 c1(C(=O)NCC(C)C)ccc2cc(C(N3CCCOC(C(C)(C)C)C3)=O)[nH]c2c1 N1(c2ncnc(NCCCCC#CC)c2C)CC2C(C(F)(F)F)CC2(CO)C1 N1(C(c2c(NCc3cccc(CC(=O)O)c3)ccs2)=O)CC2COCC2C1 CCC(CC)(CC)C(=O)N1CC2(C1)CN(C(c1ccc(Br)c(Cl)c1)=O)C2 c1(C(N2CCCCC2C(=O)NCc2cc(I)c[nH]2)=O)cc[n+]([O-])cc1 C1(C(C)C)CN(C(c2cnn(CC(F)F)c2)=O)CCC1NC(c1cccnc1)=O N1(C(C(C)CSC(F)(F)F)=O)CC(C2(NC(=O)CC3COCC(C)(C)O3)CC2)C1 c1(C(CC)O)ccc(F)cc1.C1(N)CC(CN)C1 C(C(F)(F)CCC(=O)NC1CCC(C(N)=O)C1)n1cc(C(C=C)(C)O)nn1 C(CS(=O)(=O)CC(=O)N1CCC(N(C(=O)C(C)c2cccs2)CCO)CC1)OC C1(C(N2CC(c3c(CC)nco3)C2)=O)(CO)CC(C)(C)C1.C1(C(=O)N)CC12CCCC2 N1(CC)CC(C(=O)NC2(CNC(C3CC3(C)C3CC3)=O)CCCC2)CCC1=O Cc1cc(CC(=O)NCC2(CNC(=O)CCCNC3CCCC3)CCC2)n[nH]1 c1(C(N2CCN(C(C(CC=C)N(C)C)=O)CC2C)=O)cn(C)c(=O)nc1O c1(CCC(C)NCCc2ncsc2Br)ccccc1 C1(CC)CC(C(=O)N(C)Cc2ccoc2)CCN1C(=O)CCCC1CCCO1 N1(C(=O)CCc2ccc(O)nn2)CCC2C(C1)CN2C(=O)CSC(F)F N1(C(c2c(C(C)C)con2)=O)Cc2nccn2CC(NC(=O)Cc2cscn2)C1 CN1N=CC(CC(=O)NCC(C(=O)NC2(CO)CCSC2)N(C)C)C1=O CC(C)(O)C(O)CNC(C1COCCC1NC(=O)Cc1ccoc1)=O c1(N2CCCC(OC)CC2)nc(N(c2cc3nc(C)sc3[nH]2)C)nc2c1SCC2 c1ccccc1[N+](=O)[O-].N1(C(=O)C)CCC(OC2CN(C3CC(F)C3)C2)CC1 CCC(CCCC(=O)NCCc1ccsc1)NC(c1csnn1)=O c1(C(=O)NCc2c(C(=O)NC(CCC(=O)OC)C)cccn2)c(F)cccc1F CC(F)(F)CC(=O)N1CCCCC1CC(N1CCCC1CSC)=O C(=O)(C(CNC(=O)Cc1csc(C)n1)CC(C)C)NCCC1(COC)CC1 c1(CC)cc(C(N2C(C(=O)NC(CC)CO)CC2C)=O)c(C)o1 C(=O)(C1=C(F)CN(C(=O)CCc2ccoc2)CC1)NCC#CC(C)(C)O N1(C(C2CC(=C)C2)=O)CCC(C)C1CC(=O)NCCCCCN(C)C C(N=c1nc(N2CCC3(CCCO3)CC2)c2cnn(C)c2[nH]1)C1CCN(C)C1 N1(C(c2c(C)nncc2)=O)CCCCCC1C(=O)NC(C)CF CC1(C)NC(=O)CC1C(N1CCC(NC(c2cnn(C3CCC3)c2)=O)C1(C)C)=O N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(CC(=O)Nc3cnccn3)C2)C1 N1(C(c2cc(C)on2)=O)CC(F)(F)CC1CCNC(=O)CCCNC(N)=O CC1CC(NC(=O)COC(C)(C)CNC(=O)Cn2cnnc2O)CS1 c1(CC)cnc(O)c(C(N2CCC(c3ccccc3)(CO)C2)=O)c1 N1(C(C=CC(c2ccncc2Br)=O)=O)CCN(CC(F)F)C(CCO)C1 Cc1cc(C(=O)NC(C)C(C)(C)NC(c2ccsc2CN)=O)cc(C)c1 c1(C(=O)NC(CNC(C2CCC2)=O)C2CC2)cc(C)ccc1SCC c1(N2CC(CN(C)C(C3(F)CCC3)=O)OCC2)nc(Cl)ncc1Br C=CC1CN(C(=O)CC(O)CC)CC1NC(c1cn(C)cc1C(F)(F)F)=O N1(C(C(F)=CCC)=O)C(C(=O)NCc2conc2C2CC2)CCC12CC2 c1(C(=O)NC(c2cccc(F)c2)CC)ncccc1NC(=O)Cc1ncccn1 c1(C(N2CCC(NC(CN(CCOC)C)=O)C2)=O)ccc(-n2cncn2)c(F)c1 c1(SCC(=O)NCC(C2CC2)NC(c2c(CC)sc(=N)[nH]2)=O)ccc(C)c(C)c1 CC1COCC(CC(=O)NC(C(=O)NCc2cnns2)C2(O)CCC2)O1 C1(c2nc(NC(=O)CCOC3CCCC3)no2)CC2C=CC1C2 N1(C(Cn2ccc(C)n2)=O)CCCN(C(=O)C=C2CCC(C)CC2)CC1C O=C(N=c1ccn(CCF)[nH]1)C(=O)c1cccc(C(=O)O)c1 CCCC(F)C(=O)NC1CC(=O)N(C2CN(C(=O)C=CC3CCC3)C2)C1 C1(CNC(c2c(CC)ncs2)=O)CCCCCN1C(=O)CNC(=O)C(F)(F)F C(=O)(C(C)CC(=O)N1CCC(N(C(c2ccc(Br)c(C)n2)=O)C(C)=O)CC1)OC N1(C(c2ccc(C(C)=O)[nH]2)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC1C1CC1 C12(C(=O)NC3CCC(CNC(=O)CC4CC(F)(F)C4)C3)CCCC1CC2 c1(C(=O)NC(CC(C)NC(=O)CCCN2C(=O)CCC2=O)C)snc(Cl)c1Cl N1(C(C(C)C)=O)CC2CC2(C(=O)NCC2CCN(C(=O)C(C)C)C2)C1 C(C(CC(=O)N1CCC1CNC(C1CC(O)(C(F)F)C1)=O)C(F)(F)F)N(C)C c1(C(N2C(C(N3CCCCC3C)=O)CCC(C)C2)=O)ccc2[nH]ccc2n1 n1(CC(=O)NCCCC2(NC(C=CC)=O)CC2)ccc(CO)n1.C(CNC(C)=O)N CCC(c1ccc(C)cc1)=CC(=O)N(C1CN(C(c2sc(O)nc2C)=O)C1)C N1(C(Cn2c(C)ncn2)=O)CC(=O)NCC12CCC2 C1(CCNC(=O)COC(F)(F)F)CSCCN1C(c1ncncc1F)=O.C(C)N c1(CS(=O)(=O)NCC2CCCOC2c2ccccc2)ncccc1Cl c1(COC)nc(NCc2cccnc2N)cc(N2CCSCC(C)C2)n1 N1(CC(=O)N(C)CC2(CNC(C(CCCC)F)=O)CC2)C(=O)NC(C)(C)C1=O N1(C(c2cc(C)n(C)n2)=O)CCC2CC2(NC(c2ccc3ncsc3c2)=O)CC1 C(=O)(CCN=C(NCc1ccc(C(N)=O)nc1)NCc1cnn(C)n1)NC c1(C(=O)NCC(CCCC)NC(=O)CN2CC=CC2)[nH]c2ccccc2c1OC CC1CC(C(N2CCC(C(CO)NC(=O)CCc3ccn(C)n3)CC2)=O)C(C)O1 C=C1CC(C(=O)OC)(COCC)C1.c12ccc(s1)C(=O)N(C)C2 N1(CC(N2CCC(c3n(-c4ncc(C)s4)ccn3)CC2)=O)CC(C)CS1(=O)=O O=C(CCCC1CCOCC1)NCC1CN(C(=O)CN2CSCC2=O)C1 c1(CC)ccc(Br)cc1C(=O)N(C)CCN(C)C(C1CCCC(C)C1)=O C1(O)(C(=O)N)CC2(CCN(N(CCC(C)c3cn[nH]c3)C)C2)C1.C(C)(C)(C)OC=O C1(C(=O)NCCN(C)Cc2nnc(O)cc2O)CCC(=O)N(c2cnn(C)c2)C1 c1(C(=O)NC(C(C)OC)CC(=O)NC2C3CCCOC23)cccc2ccnn12 CC(C)(CNC(=O)COC(C)(C)CNC(=O)CC1CCCO1)C(N)=O N1(C(C(=Cc2cccnc2)C)=O)CCC(CN(C)C(C2CCC(F)C2)=O)CC1 c1(C(=O)NC2C(C)N(C(=O)CNC=O)CCC2)cc2cc(Cl)sc2[nH]1 C1(NC(CC=C(C)C)=O)CCC2(CC1)CN(C(=O)CC1CCCCC1C)C2 c1(C(C)(C)C)ccc(C(N2CCCCC2CNC(C2CCCC2(F)F)=O)=O)cc1 N1(C(C2C(CC)C2)=O)CCCC2CN(C(=O)CCCN(C)C)CCC12 c1(Oc2c(C)cccc2)ncc(Cl)cc1F.N1(C(Cn2cc(N)nn2)=O)CCOC(C)C1 CCC(CC(=O)NCC1C2CC2CN1C(=O)C=CCOCC(F)(F)F)SC C(=O)(C1=NOC(C)C1C)NC(C(C)C)CCN(C)C(C1CC=CCC1C)=O C(=O)(C1=CC2CCCCC12)N1CCCC(CNC(COc2cn(C)nc2)=O)CC1 C1(F)(C(=O)NCC(C)(C2CC2)NC(c2ccc(CCC)[nH]2)=O)CC12CCCCC2 Cc1c(-c2ccco2)n[nH]c1C(=O)NCC1(NC(C2CC(CN(C)C)C2)=O)CC1 C12(C(=O)NCC3N(C(c4ccc(CC)s4)=O)CCC3)CCC(CO1)C2 c1(CCC(=O)NCc2cn(CCNC(=O)C(F)(F)C(F)F)nn2)ccc(O)c(Cl)c1 C1(C(N(CC(=O)N(C2CC(OCC)C2)C)CC2CC2)=O)CC2CCCC2C1 C(=O)(CC(C(F)F)NC(=O)CCCCOC)NCC(COC)(C)O c1(OC)ccc(C)c(C(N2CCCOC(CCNC(=O)C(C)=C3CCC3)C2)=O)c1 CC1CN(C(=O)C(c2cccc(Cl)c2)(F)F)CC1NC(=O)C(C)(C)C c1(NC2CN(C(CCOC(C)C)=O)C(C)C2)ncc(C#N)c2ccsc12 C1(C(C)C)OCCC1C(=O)N(CCC(=O)NCC(O)C1CC1)C Cc1cc(C#N)cc(C)c1CC(=O)N(CC(C)CNC(=O)CC)C CC(C(=O)N1CCN(C(=O)CN(C(=O)CC(C)(C)C(F)F)C)CC1)P(C)(C)=O Cc1cc(NCC2(C)CCCN2C(C2(c3ccncc3)CCC2)=O)nc(C)n1 CC(CC(=O)NCC(O)CNC(C1(Cc2cccc(Cl)c2)CC1)=O)C(F)F C1(NC(C(CC2(NC(C)=O)CCC2)=O)=O)CCN(CC2CC3CCC3C2)CC1.NC c1(C(N(C)CC2CN(C(=O)OC(C)(C)C)CCO2)=O)ccn2c1CCC2 CC1(C)CCN(C(c2cccc[n+]2[O-])=O)C1CC(N1CCOC(CF)C1)=O c1(OCC(=O)NCC(C)N(C(Cn2c(C)ncc2)=O)C)ccc(F)nc1 C12(C(N3CCCC(CC=C)(NC(c4ccc(F)s4)=O)C3)=O)CCC(C)(CC1)CO2 c1(C(C(=O)NCC(C)CNC(C2(N(C)C)CC2)=O)C2CCCC2)ccccc1 Cn1nccc1CCC(=O)NC1(CCCCNC(=O)C(F)n2ccnc2)CC1 Cc1ccc2c(CNCC3CCCN3C)c[nH]c2c1.C12(CCC1)CC(=O)N2 c1(C(=O)NC2CN(C(C3(F)CC3)=O)CCC2C(F)(F)F)cc2ccnn2cn1 n1(-c2cn(-c3cccc(C(=O)O)n3)nn2)ncc2cc(Br)cnc12 N1(C(CCNC(C(CC)OCC)=O)=O)CC(C)CCCC1C N1(C(C(c2ccc(F)cc2)C)=O)CC(CNC(=O)CSc2cn[nH]c2)CC(C)C1 C(C)(C1CCCCC1)=CC(=O)N(CCCNC(C(CC1CC1)OC)=O)CCO c1(C(=O)NCCSc2cn(-c3cncc(C(=O)O)c3)nn2)ccc(Cl)cc1CO N1(C(C2CCCC(O)C2)=O)CC2(C(N3CCC3)=O)CC1CO2 C1(CN(C(COCCCOCC)=O)C)Cc2cc(OC)ccc2O1 C(=O)(C1=NC2=NCS(=O)(=O)C12)NCC(c1ccccc1)CNC(CCC(N)=O)=O C(=O)(C(N)CCO)NCc1cn(CC(C)C)nn1.c12ccc(o1)CONC2=O C#Cc1ccc(Br)c(C(=O)NCCCN(C(=O)CC(F)(F)F)CC)c1 CCCCC(C)(C)NC(=O)CCCn1cc(CN(C)C)nn1 C1(CCC)CN(C(c2occc2C(C)C)=O)CCN1C(=O)C(CSC)NC(C)=O C1(C2CCCN(C(=O)Cc3cccnc3)C2)(NC(=O)CCCF)CC1 C1(F)(C(N(CCC(C)O)C)=O)CCCN(C(C2CC23CCCC3)=O)C1 N1(C(C(CC#C)(C)C)=O)C2CCC1CN(C(C1CC(C)OC1=O)=O)C2 c1(C(N2C3C(N(C(c4n(CC)ncc4)=O)C)CC(C3)C2)=O)nccc2n[nH]cc12 c1(CC)cc(C(=O)N(C)CCOCCNC(=O)C(C2CCC(=O)N2)C)on1 C1(C(=O)NCCN2CCc3ccccc32)CC2CCC1N(C(=O)Cn1cccn1)C2 c1(OC)ccc(-n2nc(-c3ccc(Cl)s3)nc2Cc2cn(C(C)C)nn2)cn1 n1(CC(N2C(CNC(CC3(OC)CC3)=O)C(C)CC2)=O)ncc(C#N)c1N N1(C(C2CCC2)=O)CCCC(N(C(=O)CC2CC(F)(F)C2)CC2CC2)C1 c1(C(=O)NCC(CC)NC(c2cc(Cl)c(Cl)s2)=O)ccc(CC#N)cc1 N1(C(CCNC(COC)=O)=O)CC=CCC1NC(=O)OC(C)C(=O)N(C)C C(=O)(C1CCCc2nn[nH]c21)NCC1(F)CC(NC(Cc2c(C)cncc2)=O)C1 CCC(C)C(CCN=c1cc[nH]cc1S(=O)(=O)N(CCC#N)C)SC C1(C(=O)NC2CN(C(C3C(=C)C3)=O)C(C)C2)CCCCC1N=[N+]=[N-] Cc1cc(C(=O)N(C)CCN(C)C(C2CC(C)C2)=O)nnc1C.C1(C2CC2)CC1 c1(-c2ccc(C(=O)NC(CC)C(=O)NC)nn2)ccc(S(=O)(=O)F)cc1 C1(CNC(C2CSC2)=O)CN(C(=O)CCCc2ccc(C(F)F)cc2)CCCO1 C1(CNC(c2cc(CC)nn2C)=O)CC(C)(C)CN1C(=O)Cc1ccc(C)cc1 c1(C(=O)NCCC2CCC(NC(C3(CC=C)COC3)=O)C2)cccc(C(F)F)c1 c1(C(=O)NC(C(C)NC(c2cc(Cl)cnc2O)=O)C)[nH]c2ccccc2c1C#N c1(C(C(=O)NC(C(C)OC)C)N(C)C)ccccc1 N1(C(c2cn(C)nn2)=O)CCCC2(CC(NC(=O)C=CC(C)(C)C)CO2)C1 C(C(=O)NCC1CCCO1)(C(C)Cc1ccccc1)N1CCC(CC)CC1 N1(C(c2cnn(C)c2)C(=O)NC(CC)(C)C)CCC(O)(c2nccn2C)CC1 c1(C(=O)NC(CN(C(=O)CC2CC(C)(C)C2)C)(C)C)ccc2c(c1)CC2 c1(NC(CC)C2CC2)ccc(S(=O)(=O)NCCC(C(F)(F)F)NC(C)=O)cc1Cl S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)N1CC2(N(C(Cc3nc(C)sc3)=O)CC2)C1 c1(CCC)cc(C(=O)NCC2(O)CC(NC(c3c(C)cnn3C)=O)C2)n(C)n1 Cc1cc2c(NC(C3CCCN3C(=O)CCc3ccccc3F)=O)ncnc2[nH]1 c1(CC(N2C3CN(C(=O)C=Cc4ccsc4)CC32)=O)ccc(F)cc1Br C(=O)(CC(C)(C)COC(C)=O)N(CC(=O)NC)C.C1(=O)C(C)(F)C(=O)O1 C1(NC(CN(C(C2CCN(CC)C2)=O)CC2CC2)=O)CCCCCCC1 N1(C(C=C(C)C)=O)CCCC(C2CCN(C(c3cn(C)c(=O)n3C)=O)C2)C1 c1(C(=O)NC2CN(C(CC(C)CF)=O)CC2CC2CC2)ccc2cncn2c1 C=C(C)CCCC(=O)N1CC(F)CC1CNC(C1CCS(=O)(=O)CC1)=O N1(C2CN(C(C(COC)C)=O)C2)CCN(C(C2(COC)CCCCC2)=O)CC1 C1(C(=O)NCC2N(C(C34OC(C)C(C3)C4)=O)CCCC2)CC2(CCCC2)C1 CC1(C)CC=C(C(=O)NCCC2CCCN2C(c2ccc(Cl)cc2Cl)=O)CC1 c1(OC)ccc(C(=O)C(N2CCC(CO)CC2C)C=Cc2cccs2)cc1I N1(C(c2cc(C(C)C)no2)=O)CCC2(CCCN(C(=O)CCOCC(F)F)C2)C1 c1(NCCCC2CC(OCC)C2)ncnc(COCOCC2CCOC2)c1C N1(C(C2(C)CCSCC2)=O)CCC2CC2(C(=O)NC2CC3(CCCC3)C2)CC1 N1(C(CC(c2nc(C3(COC)CC3)sc2)C)=O)Cc2n[nH]cc2C1C(=O)OC C12(C(=O)NCCC3(NC(c4ccc(Br)o4)=O)CC3)CCCC1C2(F)F C1(CC(N2CCC(CO)C2)=O)CCCCC1NCc1ccncc1 C(C(C)CN=c1[nH]cnc(Cl)c1Br)NC(c1c(OCCC)nc(C)cc1)=O CC1(O)CCC(C(N2CC(NC(=O)C(N)=O)C3(CC3)C2)=O)CC1 c1(OC)c(Br)cc(NC(C2CCC(NC(C)=O)CC2)=O)cc1Br c1(C(=O)NCC2(O)CCN(C(Cn3c(CC)nnn3)=O)C2)cnn2ccn(C)c12 CCC(C)C(O)C(C)C(=O)NC1CC(CCNC(C2CC2OC)=O)C1 Cc1scc(C(N2CC(C(C(=O)NC3CCN(C4CC4)C3)N(C)C)C2)=O)c1C c1(NC(C(=O)Nc2cccc(SC)n2)=O)ccnc2cccc(F)c12 N1(C(CCSCC(C)C)=O)CCN(C2CCN(C(=O)CC(C)O)CC2)CC1 CC(C)CC(C)CC(=O)NC1CCC(N(C)C(c2ccc3ncccn23)=O)CC1 c1(N2CCN(CCCCC)CC2)nc(=NC)[nH]c(=NC2CC(CC(F)F)C2)[nH]1 N#Cc1cc(C(=O)NC2C3CCC2N(C(C2CCCN2C=O)=O)C3)ccc1F CC(CC(=O)NC1CCOC(C)C1)C(C)(C)NC(C1CC2CCCC2C1)=O c1(N(CC(CN(C(C=CC(CC)=CC)=O)C)O)C)ccc2nc(OC)[nH]c2c1 N1(C(C23CCC(OC)C2C3)=O)CC2(CO)CC1(C(=O)NC1CCCCCC1O)C2 C1(CC(=O)N(CCn2ncc(C)c2)C)CCN(C(=O)CC2CCCCO2)CC1 c1(SC)nc(O)nc(C)c1C(=O)N(CCCNC(=O)CCC1CCOC1)C(C)C c1(C(N(CC(=O)N(C)Cc2nccs2)C2CC2)=O)cc(C2CCC2)nn1C CCC(C)(C)C(=O)C(=O)NC1CCN(C(c2ccn3ccsc23)=O)C(C)C1 C1(C(c2n(CC)nnn2)NCCN(C)S(=O)(=O)N(C)C)CC2(CCCCC2)C1 Cc1cc(C(=O)NCC(C)(C)NC(C2C3C(=O)OCC23Br)=O)cnc1O n1(CC)c(CC(N)C(=O)NC2CCCCC2C(=O)OC)nnc1O c1(CNC2CCC(C(N(c3cccc(C#N)c3)C)=O)C2)cc(Cl)c(O)cc1F c1(C(=O)NCC2CCCN2Cc2ccccc2)c(C2CC2)cccc1Br c1(OC)ccc2c(C(N3CCN(C(C4(CO)CCC4)=O)CC3C)=O)cnn2c1 C1(CN(CC(C)C)CC)CCN(C(=O)Nc2ccsc2OC)CC1 C1(C(=O)NC2C3(C(=O)Nc4cccc(SC)c4)C4CC2CC34)Cc2nccn2C1 CC(C)CC(C)CC(=O)N1CCN(C(=O)CCSC2CCCC2)C(CF)C1 c1(NC(N)=O)ccc2sc(OCC(=O)NC3CCOC3)nc2c1 N1(C(C(CO)NC(CN2CCC(C)CC2)=O)=O)CCC(C2(C)CC2)C1 N1(C(CC(=C=C)C)=O)CCC2(CC1)CC2(CO)CNC(C1CC1c1ccsc1)=O Cc1cc(C(=O)NCCN(C(C2CC(F)(CF)C2)=O)CC2CC2)ccc1F c1(C(N2CCCC(NC(C3C(CN(C)C)C3)=O)CC2)=O)ccc2cc[nH]c2n1 c1(CN2C(C(N(CCO)Cc3cccc(C)c3)=O)CC(C)C2)ccc(O)c(Cl)c1 C1(C(=O)NCC2CC(C(=O)NCc3ncc(CC)[nH]3)C2)CCC=CCCC1 N1(C(c2c(C)nc(C)o2)=O)CCN(C(C2CC2C(F)(F)F)=O)C(CCO)C1 c1(OC)cc(CNC(c2ccc(=O)n(C3CC3)c2)=O)ccc1Sc1ccccc1 c1(C(=O)NC2CC(CCNC(C3(C)CCCCCC3)=O)C2)ccc(P(C)(C)=O)o1 C1(NC(c2csc(C)c2N)=O)CC1C1CCCN(C(=O)COC(F)F)C1 N1(C(c2cc(C)n(CO)n2)=O)CCC(NC(c2sc(C3CC3)nc2C)=O)C(C)C1 C1(NC(C(CSC)C)=O)CN(C(=O)CCc2ccc(O)cc2)CCC12CCC2 c1(NC(=O)CC2(O)CCN(Cc3cc(I)c[nH]3)CC2)[nH]nc2ncccc12 CC(C)(CS(C)(=O)=O)C(=O)N1C2CCC1CC(CNC(=O)CCc1ccoc1)C2 C1(NC(Cc2n(C)cnc2)=O)CN(C(c2sccc2Cl)=O)C2CCCC12 c1(C(N2CCC(NC(c3ccn(C)c3)=O)(CO)C2)=O)cc(C(N)=O)cc(F)c1 c1(-c2ccc(C(C)(C)C)cc2)cc(C(F)(F)F)cc(F)c1 c1(C(N(C2CN(C(C3CCCOC3)=O)CC2(C)C)C)=O)c(F)ccc2c1OCO2 c1(OC(C(=O)NCCC)(F)F)ccc2ccccc2c1Br C(CCCCCCO)NC.c1(OC)ccccc1OCc1cn(CCCO)nn1 N1(C(C(C)Cc2ccccn2)=O)CCCC(CCNC(c2nocc2Cl)=O)C1 c1(C(=O)NC2CCC(CNC(c3ncn(CC)n3)=O)C2)cccc(Br)c1 C1(CC(=O)NC2(C#C)CCOC2)CN(C(=O)Cn2nnnc2C)CCC1C c1(C(=O)NC(C2CN(C(C3CC(S(C)(=O)=O)C3)=O)C2)C)cc2cc(F)ccc2[nH]1 CC1CN(C(C2CCS(=O)(=O)C2)=O)CCN1Cc1ccnc(Cl)c1 Cc1c(Cl)cnn1CC(=O)NC1CN(C(=O)Cc2cccs2)CC1C CC1(C)CCN(C(=O)CCc2nc(O)n[nH]2)C1CC(N1CCC(O)(CO)C1)=O c1(C(=O)OC)ccc(C)c(C)c1.C1(N2C3C(C(O)C3)CC2=O)CCC(C)(C)C1 C12(C)CC(F)(F)CN1C2=O.C1(C)CCCC(=O)N1.c1(COC)ccccc1 CC1CN(C(=O)CC(C)(C)C#N)CCC1C(=O)N(C)CC1CC(F)(F)C1 N1(C(C)C(=O)NCCC(O)CNC(c2cccnc2)=O)CCN(C)CC1 c1(CCNC(C(Cn2ccc(C)n2)C)=O)ccc(CNC(c2cnco2)=O)cc1 C12(NCc3c(O)ncc(C)c3)CCCN(C(=O)OC(C)(C)C)CCC1C2 c1(C(N2CCN(C(C(C)CC(N)=O)=O)C(CCO)C2)=O)cccc2c1nnn2C C1(C(=O)NC(c2ncc(C)o2)C)CC12CCN(C(=O)CC1(COC)CC1)C2 N1(C(c2c(C)nc[nH]2)=O)CCC(NC(=O)C(O)Cc2[nH]cnc2C)C12CC2 C(=O)(CC(C)CC(C)(C)C)N1CCC(CNC(c2cn(CCOC)nc2C)=O)C1 C(CC(C)C)(C(=O)NCC)N1CCCC(CN(CC=C)C)C1 N1(C(c2c(C)snn2)=O)CCN(C(c2ccc(=O)n(C)n2)=O)C(C(C)C)C1 c1(OC)ccc(C(C)C(=O)NC2CC(F)(CNC(=O)CC(C)OC)C2)c(C)c1 O=C(C1=NOCC1)NCCC1CCN(CCOC2CCOCC2)CC1 C1(C(C)NC(C2CC(NC(C3CC(=C4CC4)C3)=O)C2)=O)CCN(C)C1 c1(C(=O)Nc2ccccc2N2CCOCC2)cc2c(Cl)c(Cl)ccc2[nH]1 CC1CC2(CO1)CN(C(=O)CCCCNC(C1CC13CCC3)=O)C2 C1(NC(CCc2cncc(C)c2)=O)CN(C(=O)C(F)C2CCC2)CCC1F C1(CNC(C2(CCC=C)CC2)=O)CC2(CC2)CN1C(=O)C(c1ccc(Cl)s1)=O N1(CC(=O)N(CCN)Cc2ccccc2)CCCC1C1CCCC1 C1(NC(C(CC(C)C)(C)C)=O)CC2(CCCN(c3nnc(C(F)F)s3)C2)C1 C(=O)(CCCC(C)(F)F)NC1C2N(C(C(C)OC)=O)C(CC2)C1 Cc1ccc(C(=O)NC2C=CC(CNC(C3CC(C(F)F)C3)=O)C2)n1C c1(NC(C2CCN(Cc3cc(F)c(Cl)cc3Cl)CC2)=O)ccc2c(c1)CNC2=O C12CCN(CCO1)C2=O.CCC(C(F)(F)F)NC(=O)C1CC1 C1(OC)CC(NC(c2ccn(C(C)C)n2)=O)CN(C(=O)CS(=O)(=O)NC2CC2)C1 c1(CNC(C2CSC(c3ccccc3)C2)=O)ccc(-c2ccon2)cc1 C(=O)(C(O)C(F)(F)c1ccccc1)Nc1ccc(C(N)=O)cc1 Cc1ccc(C(N2CCC(C(C)(C)NC(c3cc(C#N)[nH]c3C)=O)C2)=O)c(F)c1 c1(C(N2CCCC(CNC(CC3(C=C)CC3)=O)C2)=O)cn2c(n1)C(C)CCC2 Cc1nn2cc[nH]c(=O)c2c1C(=O)N(CC(O)CNC(=O)CN1CC=CC1)C C1(CN2CC3(CC(NC(c4ncn(CC)n4)=O)C3)C2)COc2ccccc2O1 N1(CCOC(C2CCCN(C3COC3)C2)=O)C(=O)NC(C)(c2ccc(Br)cc2)C1=O C(=O)(CCN=C(NC1CC1SC(C)(C)C)N1CCC(c2cnccc2C)C1)NC N1(C(c2c(C#C)cn(C)n2)=O)CCC2CC(C1)CN(C(c1ncsc1C)=O)C2 N1(CC)CCCC(C(=O)NCC(F)CNC(c2ccc(OC)cn2)=O)C1 C(CCCCCC(=O)N1CCC(NC(c2cnnc(O)c2)=O)C1(C)C)SC c1(C(c2n(CCOCC)nnn2)Nc2cncc(C#N)n2)cc2ccc(O)nc2s1 c1(CC)cc(NC(C2CC3CC3N2C(C2CCCS2)=O)=O)cc(F)c1 c1(-c2n(C(C=C)C)nc(-c3ccncc3)n2)ccc2nnnn2c1 C#Cc1cccc(CC(=O)NCC2CCN(C(C3CCS3(=O)=O)=O)CC2C)c1 C(=O)(CS(=O)(=O)Nc1c[nH]nc1-c1cccnc1)N(C(C)(C)CN(C)C)C1CC1 Cc1cc(C(O)C)ccc1F.S(=O)(=O)(C(C)CN(C)C)N1C(C)C1 c1(CC(=O)NCC2OCCCN(C(CCC(C)(C)F)=O)C2)ccc2ccoc2c1 N1(C(CC(C(C)C)O)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccc(F)cc1F N1(c2ccnc(NCC(N3CCCCC3)C)n2)CC2CS(=O)(=O)CC2C1 c1(C(N2C(CNC(Cn3c(C)cc(C)n3)=O)C=CC2)=O)csc2c(Cl)cccc12 CC(C)(C)CC(O)C(=O)N1CCCC1C(=O)NCc1cn(C2CC2)cn1 c1(C(=O)NC(c2cc(F)ccc2F)CC(=O)OC)ccnc(OC)c1F N1(C(C2C(OC)CCC2)=O)CC2CN(C(=O)Cn3ccnc3C)CCC12 CCC(C)(C)CC(=O)N1C2CCC(C2)C1CC(=O)NCCOC1CCOC1 Cc1cc(CN2CCC(NC(c3nc(C)c(C)nc3C)=O)C(O)C2)cc(C)c1Cl CCC(C)C(O)C(=O)NCCCN(CCCCNC(=O)C(C)C(C)(C)C)C CC(CCNC(=O)CC1CCCCO1)CCNC(c1c[nH]nc1C1CCC1)=O N1(C(C=CCOC)=O)CCC12CCCN(C(=O)C(c1ccccc1)OC)C2 C1(C(N(C2CCN(C(C34CSCC3C4)=O)CC2)CCC)=O)CC2(CSC2)C1 C1(=CC(=O)NCCC2N(C(CC3(OC)CCC3)=O)CCC2)CCC(C)CC1 C(=O)(C(O)C(C)(C)C)OCC1C(CNc2ccccc2)N(C(C)=O)CC1 C(=O)(C1=Cc2ccccc2C1)N1C(C(=O)NC(C)CCC2CCCC2)COCC1 C1(CCOC)CN(C(=O)C2=C(Cl)CC2)CCC1Nc1cc(C)nc(C)n1 c1(C(N2CC(CC)OCC2)=O)ccc(Br)cc1SC1CC1.C12(CC1)C(=O)NC2 C1(CC)CCN(C(=O)C(=O)NC)C1CN1CCOCC1C(C)C c1(NCC2N(CC)CCC2)nc[nH]c(=NCC2(OCC)CCCCC2)c1C CN1CC=CCC1CC(=O)NC1CCN(C(c2ccc(C(F)F)[nH]2)=O)C1C1CC1 N1(C(C=CC)=O)CCC(C2CC2)C1CNC(c1nc(C2CCOCC2)oc1C)=O N1(C(Cn2cc(C(C)O)nn2)=O)CC(NC(c2ccnc(C3CC3)n2)=O)CC1C CN1CCc2cc(C(=O)NCCC3(NC(=O)C4CC4)CCCC3)ccc21 C(=O)(CC1CCOc2ccccc21)NCC(C)(CO)NC(=O)CCc1cncs1 c1(C(=O)NCC(O)CO)cc2ccc(Cl)cc2[nH]1.C12CCC(CC1)CNC2=O n1(C(C)C)ncc2c(N(C)Cc3cnn(CCF)c3)[nH]c(=NC3CCC3)nc12 c1(N(C)Cc2c(C)nn(C)c2)ncnc(N2CCN(Cc3ccco3)CC2)c1C C1(C(=O)NC2(CN(C(C(C3CCOCC3)OC)=O)C)CCC2)CCC(F)CC1 C1(C(=O)NC(CCN(C(C(C)NC(C)=O)=O)C)C)CC2CS(=O)(=O)CC2C1 CCCCC(C)C(=O)NCCCOCC(=O)NCc1cnc(CC)nc1 C1(NC(CCC(=O)NC)=O)CC2CC1CN(C(=O)CC1CC(OC)C1)C2 c1(C(=O)NCCC(C)NC(=O)COCC=Cc2ccccc2)cccnc1S C(C(COC)C(=O)NCC1CCCC(NC(c2ccc(NC=O)cc2)=O)C1)OC C1(C(=O)NCC(C)OC)CC(C)(C)CCN1C(c1scnc1C)=O N1(C(COC(C)C)=O)CC2CCCN2c2ccccc21 CN1CCCC(C(=O)NCC(O)CNC(c2cc(N(C)C)n[nH]2)=O)C1 CON(CCC(=O)NCC(C)C(C)(F)F)C(=O)C1CN(C)C(=O)N1 C(=O)(CCCC(C)NC(C1CC(C)=NO1)=O)Nc1c(CC)nsc1 c1(CCC)nnsc1C(=O)NC1CCC(NC(c2scnc2Br)=O)C1 n1(CC)ncc(C(N2CC(NC(=O)CC3CCSCC3)CC2C)=O)c1Cl c1(C(N2CCCC(CCNC(c3c(C#N)nc[nH]3)=O)C2)=O)cccc2nncn12 c1(C(=O)NCCCCNC(C2C3CC4C(C3)C24)=O)cc2ncccn2n1 c1(C(=O)NC2CC(C)CN(C(C3CC(F)(F)C3)=O)C2)nn(C)c2ccccc12 Cc1cc(NC(C2CCC(NC(=O)C=Cc3ccccc3)CO2)=O)nc(Cl)c1 c1(CNCCN2CCN(C(c3n(C(C)(C)C)ncc3)=O)CC2)ccnc(Cl)c1Cl C1(C)(COC)CC(NC(=O)C=CCCC=C(C)C)CN1C(C1CC=CCC1C)=O C1(C)(CNc2cccc(CC(=O)OCC)c2)CC(OC)CN1C(=O)C=CSC c1(CCC)ccc(CNC(C)COCc2ccccc2)s1 C(=O)(C(C)(C)C1CCCN1C(C1CCC1C#N)=O)NC(c1nc(=O)o[nH]1)C c1(C(=O)NCCC(CCNC(CN(C)CC)=O)C)cn2cc(C)c(C)cc2n1 C1(C(N(C(C=C)C)CCCC)=O)CC(CCCCCO)C1.C12(CC1)C(=O)NC2 N1(C(Cc2nccc(C)n2)=O)C(C)CC2CN(C(=O)COC3(C)CCCO3)CC12 CC1CN(C(=O)CC(F)(F)C(F)F)CCCN1C(c1cnc(NC2CC2)s1)=O Cc1cc(C(=O)NCCN(C(=O)CC2CCCCCC2)C(C)C)ncc1C(N)=O c1(C(=O)NCC2C(C)(C)CN(C(c3ccnnc3S)=O)C2)cccc2[nH]ncc12 N1(NC(C2C(C)=CCS2)=O)CCc2oc(C)nc2C1.C12(CCCCC1)C(=O)N2 CCCC(C(=O)NCCCCCCNC(C1CC1c1nccn1C)=O)S(N)(=O)=O c1(C(N2CC(CNC(c3n(C(C)C)ccn3)=O)C3C2C3)=O)cccc2nsnc12 C1(F)(CNC(c2c(=O)ccn(C)c2)=O)COCCN(C(=O)C2=NNC(=O)C2)C1 C(=O)(C(C)(C1CC1)N(C)C(=O)NC(C)C)N(CCCC)CC(N)=O C(C1c2ccccc2CCN1C(c1cnc(O)s1)=O)NC(C1CCCC2CC12)=O C(=O)(C(C)CC(=O)N1CCC(CF)(NC(=O)C=C2CCCCC2)C1)OC N1(C(C(CC2CCCC2)NC(CC(C)N(C)C)=O)=O)CCS(=O)(=O)CC1 O=C(CCCC(F)(F)F)NCc1ccc(CNC(c2csc3sccc23)=O)cc1 c1(C(=O)NCCOCc2nc(C)sc2)ccccc1-c1nc[nH]n1 c1(NC(CC2N(C(c3ncn(C)c3)=O)CCOC2)=O)cccc(O)c1Br C12CC(C(C)(C)C)CN(C1)C(=O)NC2.c1cc(Cl)c(Cl)[nH]1.Cn1nccc1CC=O C1(C2CCN(C(C3CCO3)=O)C2)(NC(C2CN3CCN2CC3)=O)CC1 c1(C(=O)NC2C(NC(Cc3c(Cl)cn(C)n3)=O)CCC2)ccc(S(C)(=O)=O)[nH]1 CCCCCCCCCC(=O)NC1CCC(C(=O)Nc2cnc(N(C)C)nc2)C1 CC(CNC(=O)N(CCN=[N+]=[N-])CCO)CC(F)(F)F C#Cc1cnn(CC(=O)NC(C)C(C)NC(c2ccc(CCC)cc2)=O)c1 O=C(NNc1ccc(Cl)nc1)c1cccnc1Br c1(SC2(C(=O)NC3(CCCNC(C4C(C)(C)C4)=O)CC3)CC2)nnnn1C1CC1 N1(C(CCCCN(C)C)=O)CC2OCCN(C(=O)CCc3ccc(=N)[nH]c3)C2C1 C1(NC(C(CNC(C)=O)(C)C)=O)COC2(C1)CN(C(=O)CC1CCCCCC1)C2 C12CC3CC1N(C3)C(=O)c1cn2nn1.c1(C(=O)OC(C)(C)C)[nH]ccc1C1CC1 C1(F)(C(=O)NCC2(O)CC(CNC(c3c(CC)n[nH]c3)=O)C2)CC12CCCCC2 N1(C(c2c(O)ncc(C(C)C)c2)=O)CC2CCCC(NC(C3CC3F)=O)(C2)C1 N1(c2n(CCCOCC)c(C(C)(C)CC#N)nn2)CCC2CSCC2C1 c1(C(c2cccc(CN3CCC(c4nc[nH]n4)CC3)c2)=O)nc2ccccc2o1 c1(NC(C(=O)NCCc2ccc(OCC)cn2)=O)cnc2ccnn2c1 C1(C(=O)NCC2CC(C)(O)C2)(NC(C(C)OCCC=C)=O)CCOCC1 c1(C(N2CCOCC(NC(C(C)(O)C(F)(F)F)=O)C2)=O)csc2ccc(Cl)cc12 N1(Cc2nccc(NC(=O)OC(C)(C)C)c2)CCOc2ccc(F)cc21 C1(C(=O)NCC2(O)CCN(C(CCc3cc(C)on3)=O)C2)CCS(=O)(=O)C1(C)C c1(OCC(=C)C)ccccc1C(=O)NCC(C)(F)CNC(=O)C(F)OC(F)(F)F C1(NC(=O)CSc2cccc(Cl)c2)CC2CC1N(C(c1cccc(CO)n1)=O)C2 N1(C(=O)CSCc2ccccn2)C2CCC1CN(C(C1(O)CCOC1)=O)CC2 c1(-c2cn(CCCC(=O)NCC(=O)NC(CC)C)nn2)ccc2[nH]ccc2c1 N1(C(c2n(CC)ccn2)=O)CC2CCC2(CC(=O)NC(CC(C)C)C(=O)OC)C1 CCC(CC)CC(F)C(=O)NCCCC(C)(C)C(=O)NCc1ccc(C)nc1O Cc1ccc(C(F)F)cc1C(=O)NC1CCC(NC(=O)C2=NOCC2)C1 NC(=O)CCCC(=O)N1CC(C2CCOCC2)C1.c1cncc(F)c1 C1(NC(c2c(C)nco2)=O)CCCCN(C(c2ncc(OC(C)C)cc2F)=O)C1 C(CNC(C1(C)CSC1)=O)(CC(C)C)NC(C(CC)SC)=O Cc1cccc(Br)c1C(C(=O)NC1CCC1O)NC(C1CCCCS1)=O CC1CCCCC1C(N1CCCC(CN(C)C(c2cn(C(C)(C)C)cn2)=O)C1)=O N1(C(c2c(N)c(F)c(F)cc2)=O)CC(NC(C2CCSC2)=O)CC12CCCC2 c1(OC)cccc(CCC(=O)NCC2CCN(C(=O)CC3CCCC(C)O3)C2)c1 c1(C(=O)NCC(c2ccccc2)N(C)C(C2(C#N)CC2)=O)cnn2cccc(Cl)c12 C(=O)(NN=c1cncc(C)[nH]1)Oc1ccccc1OCSCC.CC CCCC(C)(O)CC(=O)NCc1cncc(C(N2CCC(NC(N)=O)C2)=O)c1 N1(C(CC=CCC)=O)CC(CNC(=O)C(c2cccc(Cl)c2)(F)F)C(O)C1 c1(CC)cc(C(=O)NCCC2(C(=O)NCC3CN(C(C)=O)C3)CCC2)on1 c1(C(=O)NCCC(C(C)C)NC(C=C(COC)C)=O)c(C(C)=O)sc2ccccc12 N1(C(CCC(C)(C)O)=O)CCC(NC(C2CCC(C3CC3)CC2)=O)C2(CCC2)C1 C(=O)(C1CCc2c[nH]nc21)NC1CCC(C)(NC(CCC=C(C)C)=O)CC1 C(C)(CNC(=O)Cc1ccc(C(N)=O)cc1)(C(C)C)NC(C(C)OCC(C)C)=O N1(C(c2ncn(CC)c2)=O)CCC(CC(=O)N(CCCO)C)C1(C)C C(=O)(CC(C=C)CCC)N1CCC(N(CC#C)C(c2ccc(CC)cc2N)=O)C1 CCCCCCC(=O)NC(C)(CSC)C(=O)NCCC1(COC)CCCC1 CC1(C)COC(=O)C1NC(=O)NCCNc1cncc(Cl)n1 C=CCC(F)(F)C(=O)N1CC(CC)(NC(c2cnc(N)cn2)=O)C1 C=Cn1ncc(C(=O)NCc2cccnc2C(=O)NCC(CC(C)C)OC)c1N c1(COC)ccccc1NC(=O)C(CO)NC(C1CCOC(C)C1)=O CC(C)(C)C1=NOC(C(N2CCCC2CCNC(C2CC(CC3CC3)C2)=O)=O)C1 Cc1c[nH]c(C(=O)NCC(C2CCCC2)NC(=O)CC2CN(C)C2)c1 C(C)(C)(CC(F)C(=O)N1CCc2nn[nH]c2C1)NC(CC1CCCC(C)C1)=O c1(CCC(=O)NC(C2C(C(=O)NCC(CSC)OC)C2)C)ccccn1 C1(C(N(CCC(=O)OCC)C)=O)CN(C(C2CC2F)=O)CC12CC2 c1(NC(c2c(OC)n[nH]c2)=O)ccc(NC(c2cnc(O)n2C)=O)c(C)c1 c1(CNC(Cc2cc(C)nn2-c2ccccc2)C)ccnc(Cl)c1Cl c1(CC(=O)N(CCC)CCNC(=O)C(O)CCN(C)C)cnc2c(=O)[nH]ccn12 C1(NC(CCN(C)CC)=O)CN(C(=O)Cc2sccc2C)CC2CC12 c1(OC)cc(CCC(=O)N(CC(C)NC(=O)C(C)(CO)OC)C)ccc1Cl C1(NC(CS(=O)(=O)NC)=O)CCOC12CCN(C(=O)CC(C)n1cccc1)CC2 N1(C(C2(c3ncc(C)o3)CC2)=O)CCC(N(C(=O)C(C2CCOCC2)C)C)CC1 c1(C(=O)NC(c2ccccc2Br)(C(=O)N(CCC#C)C)C)ccn2ccnc2c1 c1(C(N2CC(C)N(C(=O)CC34CCCC3C4)CC2)=O)ccc2c(n1)NCC(=O)N2 C1(CC#C)(C(=O)NC2CC(CCNC(=O)CS(C)(=O)=O)C2)CCOCC1 Cc1cc(NC(=O)CN(C(c2cccnn2)=O)C(C)C)c(O)cc1F c1(-c2ccc(C(C(F)(F)F)(F)F)cc2)ccc2ccncc2c1 Cc1ccc(Br)c(C(=O)NC2CCC23CN(C(=O)C(O)C2CC2)C3)c1 Cc1cc(C(=O)NCCCN(C(c2coc(Cl)n2)=O)C(C)C)ccc1-n1cccn1 C1(C(F)F)(CO)CCN(C(=O)Cn2cc(C(O)Cn3ccc(C(=O)OC)n3)nn2)C1 c1(C(=O)NC2CN(C(Cc3nc(C)[nH]n3)=O)CC2C)ncc(C2CC2)cc1F CC(C)(O)C(F)(F)C(=O)N1CCC(C)(CNC(=O)CN2CCC(O)CC2)C1 C1(CC(=O)N(C)CC2CCN(C(C=C(C)C(C)C)=O)C2)CCS(=O)(=O)C1 Cc1nc(C(=O)NCCC2CN(C(=O)Cc3c[nH]nc3O)C2)nn1-c1nc[nH]n1 c1(NC(=O)NCC(C)(C2CC2)NC(CN(c2cn(C)nn2)C(C)=O)=O)ccccc1 CC(CC(=O)NC1(CO)CN(C(C2CCCN2CC(F)(F)F)=O)C1)CC(C)(C)C C(=O)(CC(C)P(C)(C)=O)NCCOC1CCN(C(c2nccc(C)n2)=O)C1 c1(N(CCCO)CCO)nc(N2CCOC(c3nncs3)C2)nc2sccc12 c1(CCC(=O)NC2CCN(C(COCCCC)=O)C2)cccnc1Cl c1(C(=O)NC2(CNC(C3(C)CCCC3)=O)CCCCC2)ccc(N)c(N)c1 N1(C(c2cc(COC)[nH]n2)=O)CC2CCC1CC2NC(=O)C(C1CCCCC1)O C1(NC(c2nc(C)oc2)=O)C(C)CN(C(c2ccc(Cl)s2)=O)CC1C CCC(C)(C(=O)N1CC(F)(CNC(c2ccc(OC)c(C)c2)=O)C1)C(N)=O C(C(CC)(CC)C(=O)N1CCCC(C(C)(C)O)C1)NC(CCC(CC)OC)=O C1(CC=C)(NC(=O)Cn2cnnc2O)CCN(C(C2CC23CCC3)=O)C1 N1(C(c2ccc(OC)cn2)=O)CCC(NC(c2[nH]nnc2C2CC2)=O)C(F)C1 C1(NC(C2CC(C)(CC)C2)=O)CCN(C(C2CC(=O)NC(=O)N2)=O)CC12CCC2 C(=O)(C1=CCCOCC1)N(C1C2CN(C(C(COC)C)=O)CC21)C CN1CC(F)CC1C(=O)NCCn1cc(C(N2CCC(C)(C(N)=O)C2)=O)nn1 c1(C(=O)NC(C2CN(C(C3(CCO)CC3)=O)CCO2)C)cc(Cl)c(Cl)n1C O=C(C1CCCc2sccc21)NCCCNC(C1CCC1)C1CC1 N1(C(c2c(COC)cccn2)C(=O)NCc2ccco2)CC(C)OC(C)C1 c1(C(=O)NC2CC(CNC(c3n(C(C)C)ccc3)=O)C2)ccc(N)c(Cl)c1 C(C)(CCC(=O)N1CCCCC1CC1(C(=O)NC(N)=O)CC1)OC c1(CCC)cc(C(N2CCC(NC(=O)CC3C=CCCC3)C(O)C2)=O)cc(O)n1 C1(CC(=O)N(C)C)CCCOC1.C1(COCC)(C)CC1C(=O)N(C)CCOC C(=O)(C1=C(C)OCCS1(=O)=O)NC(CCOC)CNC(c1cscc1C)=O N#CC1=C(C(=O)NCCN(C)C2CC2)CCC1.C12CN(C1)C(=O)C1(CC1)C(=O)O2 Cc1cc(N(CCCC(C)C)C)n2ncc(Br)c2n1 c1(C(N2C(CNC(C3CC3F)=O)COCC2)=O)cc([N+](=O)[O-])c[nH]1 C1(C(=O)NCC(CC(C)C)NC(=O)C=CC2CCOCC2)(OC)CCCCCC1 C(CN=[N+]=[N-])(C(=O)N1CCSCC1)NC(Cc1cn(C)nc1)=O c1(CC(N2C(CNC(C(C)NC(C)=O)=O)CC(O)C2)=O)c(C)nn(C(F)F)c1C CCCCC(=O)NCCCOCCN(C(C12CC(O)C1C2)=O)C(C)C c1(NCC2CCN(C(C3CN(C)CC(C)O3)=O)C23CC3)ncc([N+](=O)[O-])c(=N)[nH]1 C(=O)(CC(F)(F)C(F)(F)F)N(C)CCOCCNC(=O)C(c1ccc(F)cc1)O C(=O)(CCS(N)(=O)=O)NC(C(C)(C)C)CNC(c1ncc[nH]c1=O)=O c1(CC(=O)NC(C(c2ccccc2)NC(CCNC(C)=O)=O)C)cccnc1C c1(C(=O)NC2CC(N(C(C3(CC)CCC(O)CC3)=O)C)C2)cc2cc(Cl)sc2[nH]1 c1(CC(=O)N(C(C)CCNC(=O)CC2CCCC2(F)F)C)ccc2c(c1)COC2 N1(C(C=C(C)C)=O)CCN(C(c2ccc(Cl)cc2)=O)CC1c1cn[nH]c1 c1(C(CC)C)nc(-c2cccc(OC(F)F)c2)n(-c2cccc(SC)c2)n1 C1(C(N(C(c2cn(-c3ccc(C(=O)O)cc3)nn2)C)C)=O)CCC(=O)N1C C12(CNC(C3(CN(C)C)CCCC3)=O)CCC(CC1)N(C(C1CC1C(N)=O)=O)C2 C(C1=CCCCC1)(c1n(C(CC)(C)C)nnn1)NCC(=C1CCOCC1)F Cc1ccccc1SC(C)C(=O)NCC1(NC(=O)C#CC2CC2)CCOC1 c1(CNC(=O)OC(C)(C)C)ccc(C(N2CC(N3CCNC3=O)C2)=O)o1 CCCC(CCC)CC(=O)N(CC(C)(C)C(=O)NCC1CSCCO1)C c1(C(N2CC(NC(C(C)OC)=O)C(O)C2)=O)c(N)ccc(F)c1C N1(C(C(C)NC(=O)C(C)(C)C)=O)CCC2(CC1)CN(C(=O)C(C)(F)F)C2 N1(C(C(C)(C)N(C)C)=O)CCN(C(c2ccccc2)=O)CC1 c1(NC(C)=O)ccccc1C(=O)NC12CC(NC(=O)CCCc3cnn[nH]3)(C1)C2 C(CC(C)C(=O)NCCN1CCN(C(C2CCC(N(C)C)CC2)=O)CC1)OC C#CC1(C(N2CCC3(CCCC3)C2)=O)CCN(C(=O)CCC(C)C#N)CC1 C1(CC)CCN(C(C2CCC(C)N2C(C2C3CC4C(C3)C24)=O)=O)CCO1 C1(n2ncc(NCC(C)(C)OCC)c2)CCCC(NC(=O)OC(C)(C)C)C1 N1(C(C2N(C)CCOC2)=O)CC2(CNC(c3ccn(C)c3)=O)CC1CO2 n1(C(CCC)c2cnn[nH]2)cc(CN(CCCC2CCCO2)C)nn1 c1(C(=O)NCCNC(CC2CC(C(C)(C)C)C2)=O)nn(C(C)(C)C)cc1Br Cc1cc(NC(C2(F)CCN(C(=O)CCCCCC#N)CC2)=O)cc(C#N)c1 CCC(CC(=O)OC)NC(=O)C(C1CCCC1)NC(=O)CC1CCCC1(C)C c1(C(=O)NCCC(C)N(CCC)C)oc(CNC(C2CC(O)C2)=O)cc1C N1(C(C2N(C(=O)OC)CCC2)=O)CC(NC(C2C(F)(F)C23CC3)=O)CC12CCC2 CN1CCOC(C(=O)NC2CC2NC(C2CC(F)(CF)C2)=O)C1 N1(C(C2CCN(C(C3=NNC(=O)C3)=O)C2)=O)Cc2ccccc2C1 CONC(=O)C(=O)N1CCC(C(=O)NC2CCCC2C(N)=O)C1C N1(C(CCCOCC=C)=O)C2CCC1(CNC(C1CCCC(O)C1)=O)CC2 N1(C(C(c2ccc(C)s2)C)=O)CC(NC(c2ccc(=O)oc2)=O)CC(C)(C)C1 CCS(=O)(=O)CC(=O)N1CCN(C(c2c(C)ncn2OC)=O)CC1 C(=O)(C(CC)CCCC)NC(CCCC)CNC(=O)CC(=O)OC c1(C(C)(C)C)ccc2cc(C(=O)NCC3(NC(=O)COC4(C)CCC4)CC3)[nH]c2c1 N1(C(C(C=C)(C)O)=O)CCC2(CCC(NC(=O)C(O)c3cnc[nH]3)CC2)CC1 c1(C(N2CC3C(NC(c4cc(O)no4)=O)C3C2)=O)cnc2c(c1)COCC2 C1(NC(C)=O)C(C)(C)C(NC(c2ncc(C(C)(C)C)o2)c2nnnn2C)C1(C)C N1(C(c2n(C)ncc2Cl)=O)CCN(C(C2(C)CCOC2)=O)CC12CC2 N1(C(CC2CCC(C)CC2)=O)CCCC(C2CCN(C(c3nncs3)=O)C2)C1 N1(C(Cc2nnc(C)s2)=O)CC2CC(NC(c3cn4cc(C)sc4n3)=O)CC1C2 Cc1noc2cc(C(=O)NCC3CN(C(=O)C(C)(C)CCC#N)CCO3)ccc12 N1(C(CN2CCC(C)C2)=O)CC(NC(c2cnco2)=O)C2(CCC2)C1 N1(C(Cc2ccc(C#C)cc2)=O)CC2CCN(C(=O)CC3COC(C)(C)C3)C2C1 C1(C(C)NC(c2n[nH]cc2CNC(C2C=CCCC2)=O)=O)CCC(C)CC1 C1(CC(=O)NC(c2n(C)cnc2)CO)CC(C(=O)O)N(CC2CCCO2)C1 C1(NC(c2n(CCCOC)nnn2)c2occc2Br)COC2(CCCC2)C1 C1(CCC)CN(C(c2ccnn2CCOC)=O)CCN1C(=O)CCOCCO N1(C(C=CC)=O)CCC2(CC1)CC2CNC(=O)CCc1ccc(C2CC2)cc1 C1(CNC(=O)CC2(O)CCC2)CCCCCN1C(=O)COC1CC(C(=O)NC)C1 N12CC3(CCCC3)C1C(=O)Nc1c(ncs1)C2=O.CCO.NC C12(C(=O)NCCC(C)NC(C3CC(O)C3)=O)CC(C1)S(=O)(=O)C2 C1(NC(C(C2CC2)OC)=O)CCN(C(c2ccn(C)n2)=O)C1C Cc1ccc(C(=O)NCCCNC(c2cnn3ccsc23)=O)nc1C N1(C(=O)NCc2c(C)occ2)CCCCC(CC2(Cc3ncccc3F)CC2)C1 N1(C(C2(C)CN(C(C3(C)CCC(C)CC3)=O)C2)=O)CC2(COC(C)(C)C2)C1 CC(C)(C[Si](C)(C)C)C(=O)N1C(C(=O)O)CCC12CCOCC2 C1(COC)CN(C(=O)C2CC2)CCN1C(c1c[nH]cc1C1CC1)=O Cc1ccc(F)c(CNC(C)(Cc2cccc(Cl)c2)CO)c1 c1(OC)cn(CC(N2CCN(C(C3OCCO3)=O)CCC2CO)=O)c(C)cc1=O C(=O)(CCC(CF)CF)NCCC1CCCN(C(c2c(C(C)C)scc2)=O)C1 c1(C(=O)NC2C(CNC(CCC(=O)OC)=O)CCC2)c(C)nn(C)c1C(F)F N1(C(C=CCOC)=O)CCC(CNC(c2ccc(Cl)nc2C)=O)C(F)(F)CC1 C1(C(N(CCCNC(c2ccnc(N(C)C)c2)=O)CC)=O)CCCC(C)(C)C1 CC(COc1ccccc1)C(=O)N(C1CCN(C(=O)C(C)(C)c2cccs2)C1)C N1(C(CNS(N(C)C)(=O)=O)=O)CC(NC(=O)COC(F)F)C2CCCC2C1 CC1CC(NC(=O)Cc2ccc(F)cn2)CCN1C(C1CC12CCOCC2)=O c1(C(=O)NC23CN(C(CSCCCC)=O)C(C2)C3)oc2c(OC)cccc2c1C CN1CCN(C(=O)C(F)n2ccnc2)CC1C(=O)NCCOC1CCC1 c1(C(=O)NC(C2CCCN2C(c2ccncc2)=O)(C)C)csc(-c2ccoc2)n1 C(=O)(C(O)CC(C)(C)C)NCC=CC(=O)NC1(CC#C)CCCCC1 C(=O)(C1CCCc2sccc21)N1C2(CCN(C(=O)C=CC=C(Cl)Cl)C2)CCC1 c1(C(N2C(CCNC(C(C)(C)OCC)=O)CSCC2)=O)ccc(Cl)c(C)c1 C1(CC=C)(C(=O)NC(C)(C)CN(C)C(c2cnn(CCN(C)C)c2)=O)CCOC1 Cc1ccc(S(N)(=O)=O)cc1C(=O)N(C)CCN(C)C(c1csnc1C)=O c1(C(=O)OC)cc(OC)cc(CCC(N2CCSCC2)(C)C)c1 N1(C(C2CC(OC)CN2C(c2nocc2C)=O)=O)CCC12CCN(C)C2 C#CC12CC1CN(C(c1cc(Br)cnc1Br)=O)C2 C(=O)(CCNC(=O)CC1CCOC1)NCCOCC(=O)OC.O=CC1CC1 c1(C(=O)NC2CN(Cc3cnn(-c4ccccc4)c3)CC2F)cc(F)cnc1Cl C=CC(C)(CCOC)C(=O)N1CC(CNC(c2ncccc2F)=O)OC(C)(C)C1 N1(C(c2ccc(COC)o2)=O)CCCC(N(C(=O)CCN2CCCC2)CCO)C1 C(=O)(C(CC)CCCCC)N1C(C(=O)NCCC(CC=C)(C)C)CC(C)(C)C1 Cc1ccc(C=CC(=O)N(C)CCN(C)C(c2cc(Br)n(C)n2)=O)c(C)c1 Cc1nc(CNC2CCC(NC(c3ccc[nH]3)=O)C2)cs1 Cn1nnc2ccc(C(=O)NC(Cc3cccnc3)C(=O)O)cc12 c1(NCC2(CCC)CCC2)cccc(S(=O)(=O)N(C)C)c1.c12ccsc1CNC2=O c1(-c2n(CCOC)c(N3CCC(NC(=O)C4CC4)C3)nn2)c(C)cc(C)cc1F C#CCCCCCCCNC(=O)C(C1(O)CN(C(c2cnnc(O)c2)=O)C1)F N1(C(CC(C=C)(C)C)=O)CCN(C(=O)C(N2CCC(C)C2)=O)C2(CC2)C1 N1(C(C(C)NS(C)(=O)=O)=O)CCN(C(=O)CC(c2ccc(O)cc2)=O)CC1CO C12(CC(N3CC(C)C(C(=O)NC4CC4c4ccc(Br)cc4)C3)=O)CCCN1CCC2 C1(NC(c2c(C)nn[nH]2)=O)COC2(CCN(C(C34CC(CO)(C3)OC4C)=O)C2)C1 CCCC(CCC)=CC(N1CCC(O)C1C(=O)NCC1(CO)CC(C)(C)C1)=O N1(C(C2CC(CNC(CCC#C)=O)C2)=O)C2C=CCC1CC2 c1(C(=O)NC23C(CN(C(C(COC(C)C)NC(C)=O)=O)C2)C3)c[nH]c(=N)nc1O C1(NC(CNS(NC)(=O)=O)=O)CCN(C(c2cncnc2C)=O)C(C)C1 Cc1cc(F)sc1C(N1CC2CC1C2NC(C1(CC(F)F)CCC1)=O)=O CC(=O)C(C)CC(C)C(=O)NCCn1cnc(C(N2CCn3nccc3C2)=O)c1 C=CC(CC)CC(=O)NCC1CC2(CC2)CN1C(=O)C#CC1(CC)CC1 C1(CCNC(C2C(=O)NCC2)=O)CSCCN1C(c1c[nH]ccc1=O)=O C1(O)(CNC(C(C)OCC(C)C)=O)CCCN(C(=O)CCC(N)=O)CC1 C(Cc1cc[nH]n1)(C(=O)NCC1CCSCC1)NC(CCOCCC)=O C1(NC(c2nnc(C)s2)=O)CN(C(=O)C=Cc2ccco2)CCC1C C(C)(C(O)C(=O)N(CC(C)C)CC1(Cn2cc(-c3ccns3)nn2)CC1)SC N1(C(CN(CCC)C)=O)CCCC(N(C(=O)CCc2ccc(N)cn2)C)CC1 c1(C(N2CCC(N(C)C(C3CCCC(F)(F)C3)=O)C2)=O)cccc2c1COC2 C(N=c1nc2c(Br)csc2c[nH]1)C1OCCCN(C(C(C)OCC)=O)C1 Cc1[nH]nc(C(N2CCOC(CNC(=O)C(C)(Cl)Cl)C2)=O)c1F C1(C(=O)NC2CCC(C(N3CCOC(C)C3)=O)C2)(OC)CC(C)(C)C1 c1(C(N2CCCN(C(C(CC)=CC)=O)CC2)=O)cnc2c(C#N)cnn2c1 C(=O)(C(F)C(C)(C)O)N1CCC(CN(C(c2cc(CC)c(C)s2)=O)C)CC1 CC(C)(O)C(C(=O)NCC(C)(C)OCCO)NC(=O)CC1CCSC1 Cc1c(F)ccc(N)c1C(=O)NC1CN(C(c2cccc(C)c2F)=O)C1 CCCC(CC(=O)N1CCC1C1CCC1)NC(c1ncccc1Cl)=O Cc1c(Cl)ccc(C(N2CC(NC(C3CN(C)CCO3)=O)CC23CCC3)=O)c1O c1(CC)cccc(C)c1NC(=O)CCN(C(=O)Cc1ccnn1C)CC1CC1 C1(N(C)C)COCC1C(=O)NCC1(NC(c2cc(C(C)(C)C)no2)=O)CCC1 c1(CCCC(=O)NC2CCOC(c3ccc(F)cc3)C2)ccc(F)cc1 CC1(C)CCC(C(N2CCCCC2CS(C)(=O)=O)C(=O)NC2CC(F)(F)C2)CC1 N1(C(C(CC#C)C)=O)CCCC12CCCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 Cc1cc(N2CCC(C(C)C)C2)n2nc(CO)nc2n1.C1(C(=O)N(C)C)CCS1(=O)=O C1(CC(=O)NCCOCCC)N(C(c2sc(F)cc2C)=O)CCC1(C)C Cc1cc(C)n(CC(=O)N(CC(C)N(C)C(c2[nH]ccc2C)=O)C)n1 c1(C(=O)NC23CCCN(C(CCC=C)=O)CC2C3)cccc2oc(=N)[nH]c12 CCCS(=O)(=O)CC(=O)NC(c1ccc(CN(C(=O)C(C)CN(C)C)CC)cc1)C c1(OC)cc(-c2cn(C3CCN(C(=O)C(C)n4cnnn4)CC3)nn2)cc(C)c1 N1(C(c2cc(=NC)[nH]cc2)=O)CC2CCC(C1CO)N2C(=O)Cc1coc(C)n1 Cc1nc(N2CCCC2C2(NC(c3c(Cl)cnn3C)=O)CC2)c(Cl)cc1C#N c1(C(N2CCC(NC(C3C(C)(C)CC3)=O)C2)=O)cc2ccc(F)cc2s1 c1(C(C)C)ccc(NC(=O)C(O)C(F)F)c(CNC(C2COCCO2)=O)c1 C1(C(=O)NCC(O)C(=O)NCC2COCC2O)(CCO)CCOC1 C12(NC(C3C(c4c(C)ccc(C)c4)CC3)=O)CC(CNC(=O)CO)(C1)OC2(C)C C(=O)(C1=CCCC1(C)C)N1CCC(O)(CN(C(c2c(C)snc2)=O)C)C1 N1(C(CSc2n[nH]c(=N)s2)=O)CC2CCC1C(NC(=O)CN1CCCNC1=O)C2 N1(C(c2c(CNC(c3coc(C4CC4)n3)=O)n[nH]c2)=O)CCC2CCCC2CC1 c1(OC)cc(C(=O)NCCCN(C(=O)C=CBr)C2CCCC2)cc(Cl)n1 c1(C(=O)NCC(CNC(CCCCC=C)=O)(C)O)cn2cccc(Cl)c2n1 N1(C(CCOCC#C)=O)CCN(C(c2ccccc2Cc2n[nH]c(C)n2)=O)CC1 c1(C(=O)NC2(C)CCN(C(=O)C=C3CCSCC3)C2)cc2c(Cl)cncc2s1 C(CCC(=O)NN1C(=O)NC(=O)C1C)Oc1nnn(C)c1-c1cccc(C#N)c1 c1(NC(=O)NCCC(C)CC(C)(C)C)ccc2cc(F)ccc2c1 c1(-c2n(C3C(C)OCC3)nc(C(C)(C)C)n2)cc2scc(Cl)c2[nH]1 C(=O)(C#CC1CCC2(CC1)OCCO2)NCCN(C(c1cc(C)c(Cl)s1)=O)C N1(C(C(CC)SC)=O)CCC(C)(CNC(c2cn(CCN(C)C)nn2)=O)CC1 Cc1cc(F)c(C(=O)NCC23CC2CN(C(C24CC(F)C2C4)=O)C3)cc1F c1(CN=C(NCC(c2cn(CC)nc2)O)NCC(F)F)cc(F)ccc1C c1(CC)cc(C(N2CCCC(C)(NC(=O)C3=NOCC3)C2)=O)cc(N)c1 c1(C(=O)NCC(CNC(c2ccsc2)=O)CO)n[nH]c2c1CSCC2 C1(C(=O)NCCCC(C)NC(=O)C(C2CCCCC2)F)CCOC1(C)C CCCCCCCCC(F)C(=O)NCC12CC(CC)(CN1C(=O)C(C)(C)CO)C2 C(c1nc2ccccc2s1)=CC(N1CCC2CCN(C(=O)C3=CCCC3)C2C1)=O CCC(CC)C(C(=O)NCC(=O)NCC(=O)NC1CC(CC(N)=O)C1)OC C(CNC(=O)COc1cnn(C)c1)(C(C)(C)C)NC(C(C)C1CC1)=O c1(C(N(C(C)CN(C(=O)CCn2ccnn2)C)C)=O)cccc(C(C)(F)F)c1 c1(C(N2CC(C3(NC(c4cncc(OC)c4)=O)CC3)C2)=O)cc2ncc(C)cn2n1 CCC(CC)(CC)C(=O)N1CC2C(CN(C)C(c3cnc(S)n3C)=O)C2C1 Cc1ccc2c(=NCCC3CCCCO3)[nH]c(=NC3CC4(COCCO4)C3)[nH]c2c1 CCC(CC(F)F)C(=O)NC1CC(CNC(=O)CCNC(=O)CO)C1(C)C C(=O)(C1=CC2(CCN(C(=O)CSCC(F)F)C2)C1)N1CCC(C2(C)CC2)C1 c1(OC)ccc(C)c(C(=O)NC2CC(NC(C3CC(=O)N(OC)C3)=O)C2)c1N C=C(C)C(CC(=O)NCCC1COCCN1C(c1cscn1)=O)OCC CC1(C)CN(C(=O)C(C)(C)C#N)CC1C(N1CC(C2(C)CC2)C1)=O N#Cc1cc(F)c(NC(=O)CC2CN(Cc3sccc3Br)CCO2)cc1F c1(C(=O)NCC(CC(=O)NC(COC)C(C)C)C)ccc2nccn2c1 C1(O)(CCC)CN(C(=O)C(C)(C)N(C(=O)CCCN(C)C)C)C1 C1(C(N2CC(NC(C(CC=CC)C)=O)C2)=O)CC2(COC(=O)N2)C1 c1(C(N2CCN(C(C(OC)OC)=O)C(C)C2C)=O)ccc2c(c1)CC(C)O2 c1(C(N(CC=C)CCNC(=O)C(C)OCCCC)=O)ccc(O)nc1Cl c1(CC)csc(CN2CCC2CNC(=O)CCSc2ccccc2)n1 CN1C(=O)CC(NC(=O)COC2CC(NC(=O)COCCCN=[N+]=[N-])C2)C1=O CC(C)CC(C)(CNC(c1ccccn1)=O)NC(c1cnc2n1CCC2)=O N1(C(CCCNC(C2C(C)(C)OC(=O)C2)=O)=O)CC(=O)N2CCCC2C1 N1(C(C2CN(C(C)=O)C2)=O)CC(O)C(O)C1CNC(C12CCCC1C2(F)F)=O CCC(C(=O)NC1CCCC1CN(C)C(C1CC(O)C1)=O)SC N1(C(=O)NC(c2nccs2)C)CCCC(OC2CCC2)C1 Cc1[nH]c2ccnn2c(=O)c1CC(=O)N(C1CCC(NC(=O)CO)CC1)C N1(C(C(N2CCOC2=O)C)=O)CCN(C(=O)C(C)(C)C2CCOCC2)CC(O)C1 C12(CNC(COC(C)(C)C(F)(F)F)=O)CCCC1CCN2C(c1cnc[nH]1)=O N1(C(c2nc(N(C)C)oc2)=O)CC(CNC(=O)CSCc2ccccn2)C(O)C1 N1(C(C2(NC(N)=O)CC2)=O)CC2CC(NC(C3CC4(CCC4O)C3)=O)CC1C2 CCC(=O)CCC(=O)N(CCC(=O)NC(C)Cc1cnn(C)c1)CCCO Cc1cc(C(N2CCCC(C(C)C(NCP(C)(C)=O)=O)C2)=O)cc(C)n1 N1(C(C2CC(C(F)(F)F)C2)=O)CCCC(C2CCN(c3nncs3)CC2)C1 c1(C(=O)NCCCCCN(C(=O)Cc2ccc(Cl)nc2)C)ccnc2[nH]ncc12 N1(C(C(CC=C)CC)=O)CC2CCCC2(N)C1.N(S(=O)(=O)NC)CC(=O)NCCCCC C1(CNC(C(CSC)C)=O)CC2(CO1)CN(C(C1Cc3ccncc3N1)=O)C2 c1(C(=O)NC2CCC(N(C(c3cn(CC=C)nc3)=O)C)C2)cc(O)ccc1Cl CCCCC(CC(=O)N(CCC(=O)N(CC(F)F)CCOC)OC)OC c1(C(=O)NCC2CN(C(COCc3n(C)ncc3)=O)C2)ccn2c(O)nnc2c1 C(CC(O)CC(=O)N1CCN(CC(C)(C)F)CC1)SC C1(NC(CC(C)NC(N)=O)=O)CCCN(C(=O)CSc2nc[nH]n2)CC1 N1(C(Cc2c(Br)cc(C)s2)=O)CCC(C)N(C(c2cc(C#N)c[nH]2)=O)CC1 Nc1cc(Cl)ncc1C(N1CCCC(NC(C2C3COCC23)=O)C1CO)=O C(=O)(C(C)(C)CC(F)F)N1CCC(C(C)C(=O)NC2CCC2(C)C)CC1 N1(C(C(C(C)C)n2cncn2)=O)CCC2(CCN(C(=O)C=CCF)CC2)C1 Cc1cc(F)cc(Br)c1NC(=O)C(=O)NC1CC2(CCCC2)C1 c1(-c2cn(CCC(=O)OC)nn2)nccc(C)n1.C12(CF)CN1C2=O N1(C(C2(C3CC3)CC2)=O)CC2CCCC(NC(C34CCCN(CC3)C4)=O)C2C1 C1(CNC(c2nn(C)c(Cl)c2)=O)C2CCCC1N(C(=O)CC1CCCOCC1)C2 CCS(=O)(=O)c1ccc(CN=C(NCc2cccs2)NCC2CNC(=O)O2)cc1 c1(NC)c(C(=O)NCCC(C)NC(C2(C(=O)N(C)C)CC2)=O)cccc1[N+](=O)[O-] C(=O)(CCCC(=O)N(CCC(C(C)(C)C)NC(=O)C(F)C1CCC1)C)OC N1(C(C(C)=CC)=O)CCC2(CCN(C(=O)C(C)CS(C)=O)CC2)C1 C1(NC(C2CSCCN2C(=O)CCC2CC2)=O)CCS(=O)(=O)CC1 CCC(CC(C)C)C(=O)NCC(C)N(C(=O)C(Cl)=CCl)CC C1(S(=O)(=O)N2CCC(N(CC=C)C(c3scc(C)c3Cl)=O)CC2)(CC=C)CC1 N1(C(C(CCC#C)NC(c2ccnc(C)n2)=O)=O)CCN2CCC1CC2 C(=O)(C(O)CNC(=O)C(c1cnn(C)c1)NC(=O)Cc1cnc(C)s1)OC CC1(C)CCCCC1CC(N1CC(NC(=O)C(c2ccccc2)C2CC2)C1)=O CC1(CC(=O)NC2CC(NC(C3(c4ccccc4Cl)CC3)=O)C2)CC(F)(F)C1 N1(C(COC(C)=O)=O)CCCC(F)(C(=O)NCC2CN(C)C2)C1 C(CCCC(=O)N(CC(C)NC(=O)CC1OCCC1(C)C)C)OC N#CC1(C2CCCC2)CCN(C(=O)Nc2cnoc2Cc2ccccc2)CC1 N1(C(CNC(CCC)=O)=O)CC2CN(C(c3cccn3C3CC3)=O)CC2C1 c1(C(=O)NC(CC(C)NC(c2cc(C)sn2)=O)C)ccc([N+](=O)[O-])[nH]1 c1(C(=O)NC(CCNC(CC(CCCC)CC)=O)C)cc2ccncc2c(O)n1 Cc1c(C(=O)NCCOCCNC(=O)Cn2cncn2)cnn1C(C)C N1(C(CC2CN(C(CC(COC)COC)=O)CC2C)=O)CCC(F)(F)CC1C c1(C(N2CCN(C(CC(C)n3ccnc3)=O)CC2C)=O)cc2nccn2c(O)n1 N1(CCCCOC)CCCn2nc(C(=O)Nc3ccc([N+](=O)[O-])cc3F)cc2C1 N1(C(c2c(CC)ocn2)=O)CCCC(NC(c2cc(F)ccc2C)=O)CC1 N1(C(c2c(CC)noc2)=O)CCC2(CCN(C(=O)C(C)(CC)CO)CC2)C(C)C1 C(CN=c1[nH]c(=NCc2sccc2Cl)[nH]c2c1COC2)n1cc(Br)nn1 C12(NC(CSCCCC)=O)COC(CNC(C3CC(C)CO3)=O)(C1)C2 c1(C(=O)NCCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)cc2ccsc2s1 Cc1nc2ccccc2n1CC(N1CCOCC(NC(C23CCC2CC3)=O)C1)=O c1(C(=O)NC(CC=C)CNC(=O)CC(CC)C2CCC2)cc2c(o1)CCCC2 c1(OCCC)ccc(CN2CC3CC2CN3C(C2CCC(C)C2)=O)c(OCC)c1 c1(C(=O)NCC(CNC(C(CC)NC(N)=O)=O)(C)OC)ccccc1OC c1(CN(CC(C)SC)CC(F)F)nc(=NCCCOC(C)(C)C)[nH]c2c1CSC2 C12(CC)CN(C(=O)CCc3cc(C)[nH]n3)C(CNC(c3cccc(N)c3)=O)(C1)C2 C1(CNC(C(CC)NC(C)=O)=O)CN(C(c2nccc(C)n2)=O)CCO1 N1(C(C(CCN(C)C)O)=O)CCC2(C1)CN(C(=O)CCS(N)(=O)=O)C2 Cn1cnc2c(NC3(CSC)CC3)[nH]c(=NC(CC3CC3)c3ccccn3)nc12 c1(C(=O)NCC(CC)(C)NC(C2CN(C)C(=O)N2)=O)cc2ccc(F)cc2cn1 C#Cc1nc(C(=O)NCC2(CNC(C3CCC34CC4)=O)CCCC2)cs1 CC1=C(C(=O)NC23CC(CNC(C4CSCCS4)=O)(C2)OC3(C)C)CCCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(NC(c2c(C)cn(C)c2)=O)CC1 CCCC(C)(O)CC(=O)N1CCC(CO)(CNC(=O)C=CC2CC2)C1 C1(C(C)NC(=O)CSc2nncs2)CCN(C(C2CC2C(F)F)=O)C1 C(=O)(C1Cc2ccccc21)NCC(CCC)C(=O)N1CCCC(CO)C1 C(=O)(CCC(F)(F)F)NC(C(C)NC(c1[nH]ccc1COc1ccccc1)=O)C C(CN=C(NCC12COCC1C2)NC(C)C)c1scc(COC)n1 C(=O)(C(C)C1OCCc2sccc21)N(CCCN(C(c1ccc(OC)s1)=O)C)C CC(C)CC(CNC(=O)CC1(C)OCCO1)C(=O)NCC(C)C(C)O c1(C(N2CC(C(C)NC(CNC(=O)NC)=O)C2)=O)cc(C)c2ncccc2c1 c1(CC)ccc(C=CC(=O)NC2CC(c3ccc(Cl)cc3)C2(C)C)o1 Cc1ccc(CC(=O)NCC2(O)CN(C(c3cc(C)c(N)cn3)=O)C2)c(F)c1F O=C(C1=NOC2(CCOC2)C1)NCC12CCC(CC1)N2C(c1cncc(Cl)c1)=O C(=O)(CC1=NNC(=O)C1)NC(C)C(CO)NC(=O)C(c1cccn1C)=O C1(CNC(C2(CC)CC2(F)F)=O)CC2(CCN(C(C3CC34CCCC4)=O)C2)CO1 c1(CC)cc2c(CC(N3CCCC(C)(NC(c4cc(C)no4)=O)C3)=O)csc2s1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCC(CCNC(=O)CCC1CCCO1)O c1(OC)cccc(CCC(=O)NCC2CCC2NC(=O)CSC)c1 C(C)(CCC(=O)NC1CCN(C(=O)Cn2ccc(C(F)F)n2)C1)OC C1(CC=C)(NC(=O)C=NOC)CCN(C(c2cnc(C)n2C(F)F)=O)CC1 N1(CC)CCCC1C(=O)NCCSCC(=O)Nc1csnc1OC c1(OC)ccccc1COC1CN(C(=O)CCN2CC(C(=O)NC3CC3C)C2)C1 c1(C(=O)NCC2CC(F)(CNC(=O)COCC3CCCO3)C2)cc(N)cc(O)n1 CN1CC(C)(C)CC1C(=O)NCC1CCCN(C(=O)Cc2ccccc2)C1 CC1(C)OC(=O)NC1C(=O)NC1CCC1c1cccc(Br)c1 C(N=c1[nH]nc(O)s1)C12C(C(=O)Nc3cncc(C4CCCOC4)c3)C1COC2 C(C(C)(C)C(=O)NC1CCOCC1NC(c1cnnn1C1CC1)=O)SC CC1CC(C(=O)NCCCCCNC(=O)C(C)O)CCC1C C1(NC(COCCCCOC)=O)CC(O)(CNC(=O)Cc2cc[nH]n2)C1 c1(C(C)NC(=O)CC2OCCOC2(C)C)cc(F)c(Br)cc1F C=CC1CN(C(=O)Nc2cnc3c[nH]nc3c2)CCC1CC(=O)OCC c1(OC)ccc(CCC(=O)NC2CC(N(C)C(C3CC(O)(C#C)C3)=O)C2)cc1O C(=O)(C(C)C(O)C(C)CC)NC(C(=O)NCCC(CC)(F)F)C1(C)CC1 c1(C(N2CC(O)C2)=O)ccc2c(n1)OCCO2.C(C(C)=CC(=O)NCCOCC1CC1)OC c1(C(=O)NCC2C=CC(NC(C3CCCN(C4CC4)C3)=O)C2)c(F)cccc1F N1(C(c2nn(C)c(Br)c2C)C(=O)NC)CCCC2(C1)NC(=O)NC2=O Cc1cn2nc(C(=O)N(C)CCN(C)C(C3CN(C4COC4)C3)=O)cc(C)c2n1 Cn1nc2ccccc2c1C(=O)NC(C)(C)Nc1cn(CC2CCCOC2)nn1 C1(NC(=O)Cc2cn[nH]c2)CCC12CCN(C(=O)CCc1cncnc1)CC2 c1(CNC(C2CC(CNC(=O)CC3CC(F)(F)C3)C2)=O)cc(F)c(F)c(F)c1 CC(CCCC(=O)N(C)CCOCCNC(=O)CCF)N(C)C(=O)OC(C)(C)C c1(C(=O)NCCNC(c2occc2C2CC2)=O)cccnc1C(F)(F)F C1(CNC(c2c(CC)occ2)=O)CCN(C(=O)C(C)CSC)CC1C1CC1 C1(N(C(CSCCOC)=O)C)CN(C(=O)CSc2cccc(F)c2)CC1(C)C Cc1ccccc1C(=O)NC1CCCCC1C(N1CCC(C#N)C1)=O CCC(CCCC(=O)NC(c1cccnc1)C)NC(C1CC=C(C)CC1)=O C1(N=[N+]=[N-])(C(=O)NCc2n(CCC)cnc2)CCN(C(=O)C(C)=C(C)CC)C1 C1(C(=O)NC(CC2(O)CCC2)CO)CCC(Sc2ccccc2Br)CC1 c1(CC(=O)N(CCNC(C2CCCC(OC)C2)=O)C)coc2ccccc12 N1(C(c2n[nH]c(=N)[nH]2)=O)CCC2(CCN(C(c3c(F)cncc3Br)=O)C2)C1 N1(C(C(=O)Nc2ccccc2)c2ccsc2)CCC2(C1)OCc1ccccc12 N1(CC#C)CCC(C(=O)NCC2(O)CN(C(c3cnc(OCC)cn3)=O)C2)CC1 CC1CCCNC1Cc1ccccc1.C12(C)CCN(C1)C(=O)NC2 C1(c2ccc(OC)cc2)C(C2CC2)CCN1C(=O)C(c1cccnc1)OC CC1(C)CC(C(=O)N2CC3CC(C(=O)NCCCN4CCC4)(C3)C2)=NO1 N1(C(C2CCCN(CC)C2)=O)CCCC2(CC(N(C(=O)C#CC(=O)NC)C)C2)C1 N1(CC)CCOCC1CC(=O)NCCC1CCCN(C(c2ccn(C)c2)=O)C1 CCCC(C(=O)N1CCC(NC(c2ccc(NC=O)cc2)=O)C1(C)C)S(N)(=O)=O N1(C(=O)Cc2cccnc2)CCN(C(=O)CC2CCCC2)C2(CC2)C1 CN1CC(O)CC1C(N1CCC(N(CCO)C(C2CSCCS2)=O)CC1)=O C12(NC(COC)=O)CCN(C(c3ccc(Cl)cc3F)=O)CC1C2 C1(CNC(c2ccc(C(C)=O)[nH]2)=O)CN(C(=O)C(C)N(C)C)CCC1(C)C C1(C(=O)NC2CCN(C(c3cc(O)no3)=O)C23CCC3)Cc2cc(F)ccc2O1 C(=O)(CS(=O)(=O)c1ccccc1C)N1CCC(O)(CCNC(C=C(CC)C)=O)C1 N1(c2ncc(C)cn2)CCCC2C1CCN2Cc1cccc(-c2cccnc2)c1 O=C1CCC(C(=O)NCC2CCCN2C(C2COCC2n2cccn2)=O)N1 C=CCC(C(=O)NC(C)COC)NC(c1cnncc1OC)=O Cc1c(N)ccc(C(N2CC(O)(CNC(C3CCCOC3)=O)C2)=O)c1Cl Cc1cc(C(=O)NC2CN(C(c3cccc(CC#N)c3)=O)CC2C)n(C(F)F)n1 C1(c2n(-c3cccc(OC)c3)nc(CC3CC3)n2)CC2CC(C1)CS(=O)(=O)C2 n1(CCCC)nnnc1C(C1(C)COC1)NCCC(O)C1CC1 N1(C(COCC=C)=O)CCC(C)(C)C1CC(=O)N(C)CC1=CN(C)C1 C1(CNC(C(C2CCOCC2)C)=O)CN(C(=O)COC2CCC2)C(C)(C)C1 Cc1ccc(C)c(C(=O)NCC2CCC(C)(C)CN2C)c1N C(=O)(CC(C(F)F)n1cccn1)NCC1N(C(C2C(C)(C)OCC2)=O)C1 c1(C(=O)NCC2C(NC(CCC(C)C)=O)C2)ccc2cnccc2c1 C1(NC(c2ccc(Cl)cc2Br)=O)CCN(C(C2CCOC2)=O)CC1CO C(N=c1cc[nH]c(C(=O)OC)n1)C1N(C(C(C)OC)=O)CCCC1 N1(C(C(CC)(C)C)=O)CCN(C(C2CC(F)C2)=O)C(c2cccnc2)C1 c1(C(N(C)CCNC(C2(C)CC(F)C2)=O)=O)cc(CO)n(C)n1 C1(NC(C2CCN(CC(C)C)C2)=O)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)CC1C C1(OC)CCC12CC(C(=O)NCC1CN(C(c3ccncc3F)=O)CCO1)C2 C(CC(C)C)(C(=O)NCCC(C)(O)C1CC1)N(C(CC1ON=C(C)C1)=O)C C(=O)(C1=NNC(=O)CC1)NCC1C2(CN(C(C(C)NC(CC)=O)=O)C2)C1 C1(NC(c2ccc(-n3cccn3)cc2)=O)COCCN(C(c2cscc2F)=O)C1 C1(NC(C2(C(N)=O)CCCCC2)=O)CCN(C(C2CC2(Cl)Cl)=O)CC(O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)NS(C)(=O)=O)ncc(F)cc1F N1(C(c2ccc(C=C)s2)=O)CC(NC(C2CC(C3CC3)=NO2)=O)CC(C)C1 c1(OC)ccc(C(C)(C)Nc2nnc(C3(C)CC3)o2)cc1 c1(C(=O)NC(C)Cn2cc(C3(O)CCOC3)nn2)ccc(OC(F)F)cn1 c1(C2C(C)C2)ccc(OC(CC)C)cc1.C(C)(CC1CCC1)N1C(=O)N1.OC c1(CC(=O)NCC2C3CN(C(=O)CCCCCF)CC23)nsc2ccccc12 C12(C(=O)NCC3CCCCN(C(c4cncs4)=O)C3)CC1Cc1c[nH]nc12 c1(C(N2C(CNC(c3cccc(C(F)(F)F)n3)=O)CC2)=O)c[nH]c2cccnc12 C(C)(CCN=c1[nH]c(-c2ccccc2)cs1)N(CCCC)CCCC c1(NC(C(=O)NC2CN(C(CCc3cc(C)on3)=O)C2)=O)ccc(Cl)cc1 N1(CC)CCN(C(=O)CC2(CNC(c3cnnn3C(C)C)=O)CC2)CC1=O c1(SCC)ccccc1C(=O)NC(CO)C(C)NC(=O)C(C)CN(C)C CN1CCC(N(C(c2cnc(C3CC3)s2)C(=O)NC2CCOCC2)C)C1 Cn1ncc(C(N2CCC(OCC(=O)NC(c3cccnc3)CO)C2)=O)c1N Cc1coc(C(N2CC(CN(C)C(c3nc(O)sc3C)=O)C2)=O)c1C CC1=C(C(=O)NCCCN2CCC(NC(=O)Cc3ccc(C)cc3C)C2)CCO1 C1(C(N(CCC=C)CCOC)=O)CN(Cc2cc(Br)ncc2Br)CCC1O c1(COC)ccc(C(N2CC(O)(C(C)NC(=O)CCNC(=O)OC)C2)=O)cc1F C1(OCC)CC2CN(C(=O)C(Cc3cc[nH]n3)NC(=O)Cn3cnnc3O)CC12 CC(CC(C)(C)C)C(=O)N1CCC(n2cc(C(C)(C)Sc3ccccc3)nn2)C1 Cc1ccc(CNC2CCN(C(c3ccc(C(F)(F)F)cn3)=O)CC2F)c(Br)n1 C12(CNC(=O)NC)CC1CN(C(C1CCC(NC)CO1)=O)C2 c1(NC(C)=O)ccc(C(=O)Cc2nocn2)cc1.C(CCCCCO)NC(C)=O C1(C(N(CC(CN(C(=O)CC2(CO)CC2)C)O)C)=O)CN2CCN1CC2 C(=O)(C1=CCC(C)(C)CC1)N1CCC(=CCNC(C(COC)N(C)C)=O)CC1 CC1CCC(=CC(N2CCCCC2CCNC(=O)CCOC2CCOC2)=O)CC1 C(=O)(C(=O)CC(C)C)NCc1oc(C(N(CCCCC)C(C)C)=O)c(C)n1 Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CN(C(C2(C)CCCO2)=O)CC1O c1(C(=O)N)ccnn(C)c1=O.CC(C)C(CCNC(C1(N(C)C)CC1)=O)CCC C(CCCCC(=O)N1CCN(C(=O)CC2CCC(C)(C)O2)CC1)N(C)C c1(CC)nc[nH]c1C(=O)N(CC(C)N(C)C(C1(CCOC)CC1)=O)C N1(C(C2C(=C)CC2)=O)CCC(O)(CCCCN2CCCCC2)CC1.C(=O)(C=C(C)Cl)N C12(C(=O)NCC(C)(C)NC(c3ccc(CC)o3)=O)CCC(CC1)OC2 N1(C(c2n(CC=C)ccc2)=O)CC2CCN(C(c3cc(F)c(C)cc3Cl)=O)CC12 N1(C(c2n(C)ncn2)=O)CCC(C2CC2)C1CNC(=O)CCC(C)(F)F C(=O)(C(C)C(F)(F)C(F)F)N1CC(=C(Cc2cnoc2)F)C1.CC1(CC)N=N1 c1(C(N2CC(CNC(c3ccc(SC(C)C)cc3)=O)C2)=O)cccc(F)c1F CC1CCN(C(=O)CCC2CCCC2)CC1NC(C1(F)CCCCC1)=O CC1(C)CCN(C(=O)C(F)CC(C)(C)NC(C2CCSC2)=O)CC1CO C(=O)(C(O)CCNC(C1(C)CCC1)=O)NCC1(CC)CCCO1 c1(N2CCC(C(C)NC(c3c[nH]c(C(N)=O)c3)=O)C2)ncnc2scnc12 Cn1cc(C(=O)NCC2CC(O)CN2C(C2CC2C(F)(F)F)=O)c2ccncc12 C1(C(=O)NC2CN(C(=O)C3CC3)C2)(CC)CCCN(C(c2cc(C)no2)=O)C1 C1(C(=O)NCCOCCN(C)C(c2ccco2)=O)C2CCC(F)(F)C12 C=CC(C)(CCOC)C(=O)N1CC(CN(C(=O)CNS(C)(=O)=O)C)C2(CC2)C1 Cc1nnccc1C(=O)NCCOC1CCN(C(=O)CC2CCCO2)CC1 CC1=NOC2(C1)CC(C(=O)NCC1COCCN1C(c1cc(C)sc1C)=O)C2 C(=O)(CS(=O)C(F)(F)F)NC1CN(C(c2ccc(OC)c(N)c2)=O)CC1C Cc1c(C(=O)NC2CC2CNC(C2CC2[N+](=O)[O-])=O)oc2ccccc12 c1(C(C)C)nn(C)c2sc(C(N3CC(NC(C4(C)CCCC4)=O)C(O)C3)=O)cc12 c1(C(=O)NCC2C(C)CCN(C(C3(CC#C)CC3)=O)C2)cncc2nnn(C)c12 C(CC1=CCOCC1)NC(C1(OC)CCC1)=O.c12n[nH]cc1C(=O)NC2 C(=O)(C(O)CCC(C)C)NCC1(NC(Cc2c(C)noc2C)=O)CCOC1 CC1CCSCCN1C(C1CC(C)(C)CN1C(=O)CCCC(=O)C1CC1)=O C1(CNC(CNC(COC)=O)=O)CN(C(c2cscn2)=O)CC(c2ccccc2)O1 C(=O)(C1=CC(O)CCC1)N1CCC(O)(C(C)NC(c2n(C(C)C)ncc2)=O)CC1 N1(C(c2nc(CCC)oc2)=O)CC2(C(N3CC(COC)C4(CC4)C3)=O)CC1CO2 CC1CCC(CN(C=O)CC(=O)N(C)Cc2cccc(I)c2)CC1 c1(C(N2CC(NC(C(C)C(F)(F)F)=O)(CO)C2)=O)cccc2nc(CO)[nH]c12 C1(C(N2CCC(C)(CCNC(CNC(=O)OC)=O)C2)=O)Cc2cccc(F)c2O1 C(C)(C(=O)N=c1[nH]nc(Br)s1)N1CC(C)N(C)C(C)C1 c1(C(=O)NC(C2CN(C(CCOCCCOC)=O)C2)C)ccc(C)c(O)n1 c1(C(N2CC3C(C(=O)Nc4ccc(OC)cc4F)C3C2)=O)c(Br)cc(Br)cc1Br C1(NC(c2n(C)ccn2)=O)CN(C(=O)CC2CC3C=CC2C3)CC2(CC2)C1 c1(C(=O)NC2(C3N(C(C(C)CF)=O)CCC3)CC2)nc(C2CC2)ncc1Cl C(=O)(C1=CCS(=O)(=O)C1)N(C1C(Cn2cc(C3(C)COC3)nn2)CCC1)C1CC1 C1(C(N(CC)C)=O)N(C(=O)CC2CCOC2)CC12CCCC2.c1(C)cocn1 Cc1ccc(Br)cc1C(=O)NC1CCN(C(C2CN(C(N)=O)C2)=O)C1C C(N=c1nc2c(cnn2C(C)C)c(NC2CC3CCCC23)[nH]1)C1(C=C)CCOCC1 c1(C(C(=O)NCCN(CCC)C(c2cc(CC)[nH]n2)=O)C2CC2)ccc(F)cc1 C12(CNC(C3C(C)C3)=O)COC(CNC(=O)CCC3CCCCC3)(C1)C2 N1(C(C2C(CCOC)C2)=O)CCC(NC(=O)C(F)(F)CN(C)C)CC1 N1(C(C(N2CCCC(NC(CCC)=O)C2)=O)=O)CCS(=O)(=O)N2CCOCC12 c1(C(N2CCN(C(Cn3cc(CCCCCC)nn3)=O)CC2)=O)ccc2nonc2c1 C1(C(=O)NC(C=CC(N2CC(CC(=O)OC)C2)=O)C)CCCC1C(C)C C1(CS(=O)(=O)NCCc2c(C)nco2)C(C)(C)C1(C)C C1(C)(CCNC(c2ccc(OC)s2)=O)CCN(C(c2noc(C3CC3)c2C)=O)C1 N1(C(CCN(C(c2n(C(C)C)ccn2)=O)C)=O)CCCC2CN(C)CC12 C1(NC(c2nc(C)oc2)=O)CN(C(C2CC(=O)NC(=O)C2)=O)CC2(CC2)C1 c1(NC(C23N(C(c4[nH]cc(C#N)c4)=O)CC(C2)C3)=O)cc2c(s1)CCC2 C1(C(C)C)CN(C(C2CN(C(=O)Cc3ccco3)CC2(C)C)=O)CC(=O)N1 N1(C(C(C)=C(C)C)=O)CC2CCN(C(c3ncc(Br)cc3C)=O)CC(C2)C1 Cn1cnc2cc(CC(=O)NCC(C)(O)CNC(=O)CC34CCCC3C4)ccc12 Cc1nc(C(=O)NC2COCC2CNC(c2cnc(N(C)C)nc2)=O)cn1C CC(C)C(C(=O)NC(C(=O)NCC1C(C)(C)C1(C)C)C1CC1)C(C)C c1(C(N2C(C(N(CC(N3CCCC3)C)C(C)C3CC3)=O)C=CC2)=O)c(Cl)cnn1C C1(COC)CC(CNC(c2ncccc2O)=O)N(C(c2cnn(C(C)C)n2)=O)C1 n1(CC(=O)NC2(CC=C)CN(C(C3(C)CCCO3)=O)C2)cc([N+](=O)[O-])nc1C C(=O)(C(F)(F)CC1CC1)NC1CC(Cn2cc(CC(COC)O)nn2)C1 C1(C(N(C(CC#C)C)C)=O)CCN(C(=O)C2CN(C)CCO2)O1 c1(CC)cc(-c2cnc(C(=O)NCCc3cccc(O)c3)cc2C)ccc1F C=CCCCC(=O)N(C1CCCN(C(c2cc(C(C)CC)no2)=O)C1)CC C1(NC(C=CC)=O)CC12CCC(NC(c1nc(CC)ncc1Cl)=O)CC2 C(C1CCCN1C(C1C2(CC2)C12CC2)=O)=CC(=O)NCC(C)(O)C1CCC1 n1(C(C)C)cc(C(=O)NCC2CC2NC(=O)C=CC(C)(C)C)c(Br)n1 Nc1ccc2c(c1)CCN(C(=O)Cc1ccsn1)CC2 c1(NCCCN(C(=O)C=CC(F)F)Cc2ccccc2)ncnc2cnccc12 n1(CC)c(C)cc(C(N2CCC3(NC(C45CC(C)(C4)C5)=O)CC3C2)=O)c1C CC(O)C(C)(C)C(=O)N1CC(NC(C2CC(=O)NC(c3cnn(C)c3)C2)=O)C1 C1(C)(COC)CC(NC(c2ccnc(O)c2F)=O)CN1C(=O)C(=O)NC1CC1 C1(C(=O)NCC2(C(N)=O)CN(C(c3cc(CC)[nH]n3)=O)C2)CCSC(C)C1 CCC(C)C(O)CC(=O)N1CC(C(=O)NC2(CCO)CCC2)C(F)(F)C1 c1(C(N(CCCCN(C(COCCC=C)=O)C)C)=O)cc(F)ccc1OCCOC S(=O)(=O)(c1ccccc1Cl)NCC(=O)NC1C(NC(C2CC(=C)C2)=O)CCCC1 c1(OC)ccc(CNC(N2CCC2C2CCCC2)=O)cc1F c1(OCCOC(C)C)ccc(-c2nc(C3CCCN3C)no2)cc1[N+](=O)[O-].C1CO1 c1(C(=O)NC2CCN(C(c3c(Cl)ccc(C)c3)=O)CC2C)ncnc2ccsc12 C(=O)(C1OC(=O)c2ccccc21)N1CC(F)CC(NC(C(C)OC)=O)C1 CCC(CCC(=O)NCC1(C)CCCN(C(=O)Cc2ccccc2Cl)C1)OC C(=O)(C(C)(C)C(=O)N1CCC(N(C(=O)CNC(=O)CC(F)(F)F)C)C(C)C1)OC C=CCCN=C(NCC12CC(CO1)C2)NC1CCCC(O)C1 c1(C(N)=O)cc(NC(c2cncc(NC(c3cnsn3)=O)c2)=O)ccc1F C1(CCC(=O)Nc2ccn(CCN(CC)CC)c2)CCCCN1C C(C)(C)(C(=O)NCC(O)CNC(=O)C(C)Sc1ccccn1)SC c1(C(=O)NCC2CCN(C(CN(C)C)=O)CC2CO)ccc(S(N)(=O)=O)cn1 Cc1coc(C(=O)NCc2ccccc2CN(C)C(c2ocnc2CO)=O)c1C C1(NC(=O)CCF)CCN(C(c2coc3c2COC3)=O)CCC1(F)F Cc1nc(C)c(CC(=O)NCC(O)CN(C)C(c2oc(CO)cc2C)=O)c(O)n1 c1(C(=O)NC(C(C)C)CCN(C)C(c2c[nH]c(Br)c2)=O)ccc(F)c2ccsc12 C(=O)(C(O)C(F)(F)F)NCC(=O)N(C)Cc1cccc(O)c1 Cc1cc(NC(C2Cc3cc[nH]c3C2)=O)cc(F)c1F N1(C(c2cn(CCOC)nc2)=O)CCOCC(F)(CNC(C2CCCOC2)=O)C1 CC(C)(C)C(O)CC(=O)NC1C2CN(C(=O)CCc3cccnc3)CC12 C1(CNC(=NCCC)NCCCN2CCCOCC2)Cc2ccccc2C1 N1(C(C(Cn2ccc(C)n2)C)=O)CCC2(CCCCC2NC(=O)C(C)O)C1 c1(OC(C(=O)NCC(CNC(c2cnn(C)n2)=O)CO)(C)C)cccc(Cl)c1 c1(C(=O)NC(c2ccc(F)cc2Cl)CC(=O)OCC)ncn2ccc(C)cc12 Cc1ccn(C)c1C(=O)NCCC(O)C(=O)N(C(C)CCC(C)C)C Cc1cn(C)nc1C(=O)NC(C)CCN(C)C(c1cc(Br)nn1C)=O N1(C(CCCOC)=O)CCCC2C1CCCCN2C(c1scnc1Cl)=O CC1CN(C(c2ncccc2Cl)=O)CC1NC(=O)C(c1ccc(O)cc1)C CCC(C)CCCC(=O)N1CCCC(O)C1C(N1CC2(C)CC1CCO2)=O c1(CC(N2CC(NC(c3ccco3)=O)C3C2C3)=O)ccc2[nH]ccc2c1 Cc1cc(C(N2CCSCC2C(=O)Nc2nnco2)=O)cc(C)c1O N1(S(CC)(=O)=O)CCCC1C(=O)NC(C)(C)CN(C)C(C1CSCCS1)=O C1(CCCNC(CC2(C=C)CCC2)=O)CCCCN1C(=O)CNC(C)=O N1(C(CC2C(NC(=O)CCc3cncs3)CCCC2)=O)CCN2CCCC2C1 C(=O)(C1Cc2ccccc21)NC1CCC(N(C(=O)CCc2nc[nH]n2)C)CC1 C(c1ccc2ncccc2c1)=CC(=O)NC1CN(C(C2C(C)(C)C2)=O)CC(F)C1 CC1CCCc2c(C(=O)NC(CNC(c3ncn4ccccc34)=O)CO)cnn21 c1(CN2C(C(=O)NCc3ncon3)CC3CC32)ccnc(F)c1Cl c1(CCC(N2CC(O)(CN(C(=O)CC3CCCN3C)C)C2)=O)ccccc1O N1(C(COCc2cc(C)on2)=O)CCC(c2cn(Cc3nn(C)cc3C)nn2)CC1 c1(OC)cnc(Cl)cc1C(=O)N(C1CCC(NC(=O)C2=CCCC2C)CC1)C CCCCC(C(=O)NCC1(Cl)CC1(F)F)NC(=O)C(C)OC C1(NC(=O)CC(F)F)CC12CCN(C(=O)CC1CCSC1)CC2 N1(C(=O)OC(C)(C)C)CC(C(=O)OCc2ccccc2Cl)C2CCCC12 C1(CC(=O)OC)CC2(CO1)CN(Cc1csc(-c3ccccc3F)n1)C2 C(=O)(CCCC(C)(C)NC(c1csc(C#N)c1)=O)NC1CN(C(C)C)C(=O)C1 S(=O)(=O)(CC(=O)N1CCC(CC(=O)Nc2ccccc2C(F)F)CC1)NC Cc1ccc(C)c(C(=O)NCCC2CN(C(C3CCC(O)CC3)=O)CCO2)n1 N1(C(C(C=C)(C)CC)=O)CC2CN(C(=O)Cc3ccc(F)c(Cl)c3)CC2(C)C1 c1(CCC)cccc(Cn2cc(-c3ncc(C)o3)nn2)c1 Cc1cncc(C(N2CC(C)(NC(C3CC4(CCC4)C3)=O)C2)=O)c1C C(=O)(CCC(CF)CF)N1CCC(C(NOCCC(NOC)=O)=O)CC1C c1(CN(CCCNCC)CC=C)c(OC)ccc(C(=O)O)c1Br C1(C(=O)NC2C(C(C)C)OCC2)CC(O)CN(C(C)=O)C1 C12CCN(C1)c1nnc(o1)C(=O)N2CCCC.C(N)(=O)NC C1(C(N(CCN(C(CCCC(N)=O)=O)C)C2CC2)=O)Cc2ccncc2C1 C1(C(F)(F)F)(OC)CCN(C(c2ccn(CCCF)n2)C(=O)NC2(C)CC2)C1 N1(C(C2CC3CN(C(C4(CCC)CCC4)=O)CC2C3)=O)CCN2CCOCC2C1 c1(-c2cc(CNc3cc(OC)ncc3C(F)F)ncc2)ncc2ccccn12 C1(CCNC(=O)C(C2CCOCC2)O)COCCN1C(=O)Cc1cc[nH]c1 c1(N2C(C(=O)Nc3ncc(C)nc3Br)CNCC2)ncnc2cnn(C)c12 C1(CNC(c2ccc(C(=O)OC)o2)=O)CC(OC)CN1C(=O)CN1CC2CC2C1 c1(C(N2CC(O)(CCNC(C(CC=C)CC=C)=O)C2)=O)cc(F)c(Cl)c(N)c1Cl c1(C(N2C(C)CCC(NC(=O)CNC=O)C2)=O)cc2cc(Br)ccc2o1 c1(C(N(C(CNC(C=CC(C)C)=O)C)C)=O)ncn(-c2ccccc2)n1 N#CCCC(=O)NC1CCC1CNC(=O)CC1CC1(Cl)Cl C1(NC(=O)C2=CCOC2)CS(=O)(=O)CC1NC(C1(c2ccccc2)CC1)=O c1(C(N2CC3CC(NC(c4c(C)ocn4)=O)C3C2)=O)ccc(F)c2ccncc12 C(CCCCCCc1ccccc1)(c1nnnn1CCCF)NCC(C)CO CC(C(F)(F)F)NC(=O)C=CCC1(NC(C2C3CCCC23)=O)CCC1 N1(CC)CCCCC1C(N1CCOC(CCCNC(C2COCCO2)=O)C1)=O Cc1ccc2[nH]cc(C(=O)C(C#N)C(=O)NC(c3ccccc3)CCO)c2c1 C12(C(N3CC4C(CNC(C(COC)(C)C)=O)(C4)C3)=O)CCC(C1)OC2C S(=O)(=O)(c1ccc(NCCN2CCC(N(C)C)CC2)c(Br)c1)NC1CC(OC)C1 CC1CCN(C(=O)CCc2cc[nH]n2)CC1CNC(C1OCCCO1)=O c1(C(N2CCC(N(C(COC)=O)C)C2)=O)cc(C(N)=O)ccn1 N1(C(=O)Cc2cc(F)cc(F)c2F)CCC2(CC1)CCN2C(C1CCCS1)=O CC(C)C(C(=O)N1CCC(C2N(C(c3cc[nH]n3)=O)CC2(C)C)CC1)N(C)C N1(C(C2C(OCc3ccccc3)C2)=O)CC2CC1C2NC(C1CCCN1CC)=O c1(C(=O)NC2CC23CCC3)cnc(C(F)(F)F)nc1 c1(C(C(=O)NCC)N(C(CC2CC=CCC2)C(=O)OC)C)cnc2cnccn12 C1(C)(C(=O)Nc2ccc(C)nc2)Cc2ccc(C)cc2C(=O)O1 N1(C(c2cccc3c2CCCC3)=O)CCCC2(CCCN2C(C2CC=CC2)=O)C1 c1(C(N2CC(N3CCN(S(CC=C)(=O)=O)CC3)C2)=O)cccc(C)c1O c1(C(N2CCC(NC(C(COC)C)=O)C(C)C2)=O)cc([N+](=O)[O-])cnc1N C(=O)(C(CN(C)C)C(C)(C)C)NCC(CCC(C)C)NC(=O)CC(O)C(C)(C)C N1(C(CCC2CCN(C)C2)=O)C2CCC1CC(N(C(=O)C#CC1CC1)C)C2 c12ccccc1C(C)N2.N1(C(N(C2CC2)CC)=O)CC(F)(F)CC1 Cn1nc(C(=O)NC2CCCC(CNC(=O)CCCOC(C)(C)C)C2)cc1F CC(C)C(C(=O)N(C)C)NC(C1CC(C(=O)OCC2CC2CO)C1)=O c1(CC)nn(C)cc1C(=O)NC1CN(C(=O)C(C)c2cccs2)C1 [nH]1nc(C2C(C)C2)nc1-c1cn(C2CCC2)nn1.CO c1(OC)ccnc(C(=O)NCCC2CCCN(C(C3(C(N)=O)CCC3)=O)C2)c1 C1(OCC(=O)NCCCCN2CCCC2)CCN(C(c2ccc(CO)s2)=O)C1 c1(CCC)cc(CN=C(NCCN2CCCCC2)NC(C)COCC)ccc1F c1(CCC)cc(NC2(CO)CN(C(c3cccnc3)=O)C2)nc(Cl)c1 C#Cc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cnc(Cl)c(Br)c1 CC(C(=O)NNc1cccc(C(F)(F)F)n1)N1CCC(O)C2(CC2)C1 C1(C(=O)NCCC)CCN(C(=O)COc2ccn(C)n2)O1 c1(NC(C(C)NC(C#C)COC)=O)ccc(C)o1 CC1CC(C(=O)NCCN(C(=O)CCNC(c2cccc(Cl)c2)=O)C)C1(C)C C(=O)(C(C)(F)C(=O)N(CC(C)NC(=O)CCc1ccccc1F)C)OCC Cc1ccc(-c2cc(C(=O)N(C)CCN(C)C(C3CC3(F)F)=O)on2)cc1 C(=O)(CC(C)(C)C(C)(F)F)NC1C(CNC(C(CCC)C(C)C)=O)C1 C1(C(=O)OC)CC(CC(N2CCC(N3CCC(C)CC3)C2)=O)CN(C(C)=O)C1 N1(C(C(C=C=C)C)=O)CCN(C(c2cc(C)nn2CC)=O)C(c2ncc[nH]2)C1 N1(C(c2ccc(C)cc2F)=O)CCC2C1CCCN2C(c1cc(Br)ccc1F)=O c1(CN(C(C)C(=O)OC)CC)nc(O)c2cc(-c3ccccc3)ccc2n1 C1(NC(C(CC2CCCC2)NC(C=CCC)=O)=O)CCNC(=O)C1 c1(C(C)NC2COC(C)(C)C2)cc(Cl)cc2ccsc12 c1(CNC(C2(F)CCN(C(C3CCC(CC)O3)=O)C2)=O)c(F)cncc1F Cc1ccn2ncc(C(=O)NC3CC(NC(=O)Cc4sccc4Cl)C3)c2c1 C1(CCCC(C)(C)C)CCCCC1.CC(C(=O)O)ONC=O c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2CC2)cc(F)c(O)c(Br)c1 C(CC(=O)NC1CC(N(C)C(C)=O)C1)(OCC)NCC=CC(C)(C)OCC N1(C(c2c(C)cccc2)=O)CC(NC(=O)CCCn2cccc2)CC1(C)C N1(C(C(=O)NCCC)C)CC(NC(c2ccnn2CCC)=O)C(C)(C)C1 C1(n2cc(CC(OC)OC)nn2)C=CCC(C(=O)NCC(C)(C)C(C)C)C1 N1(C(C=COCC)=O)CCCCC1CCN(C(=O)C=CCCc1ccccc1)C C1(C(C)NC(=O)CC2CCCCC2)CCN(C(=O)CCNc2csnn2)CC1 C1(O)(C(=O)NCC(C)NC(=O)CCCn2ccnn2)CCCC(C)(C)C1 c1(OC)cc(C(N2CC3CC(C2)C3NC(c2nnc(O)nc2O)=O)=O)c(Cl)cn1 C1(CNC(c2c(C)ccnc2)=O)CCN(C(c2cc(C#N)oc2C)=O)C12CC2 c1(C(N2CC3CCCN(C(C4C(=C)CC4)=O)C3C2)=O)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NC23CN(C(C(C(C=C)C)C)=O)C(C2)C3)ccc(C)c([N+](=O)[O-])c1 N1(c2cc(CC(C)C)ncn2)CCC(NC(c2n[nH]c(C3CC3)n2)=O)CC1C c1(C2(C)COC2)nccc(=NC=O)[nH]1.C(CCC(F)(F)c1ccccc1)NC c1(OC)ccc(CCN=C(NC2CCSCC2)NC2CC(OC(F)F)C2)cc1O N1(C(c2csc(C)c2N)=O)CC2C3CCC(C2C1)N(C(C1(NC(N)=O)CC1)=O)C3 C1(CC(=O)NCC2CCN(C(c3c(C)scn3)=O)C2(C)C)OCCOC12CCC2 Cc1cccc(CC(=O)N(CCC(C)(C)NC(C2CCCC(C)(C)O2)=O)C)c1C CC(CS(C)(=O)=O)C(=O)NC1CCC(NC(=O)Cc2cnn(C)c2C(F)F)C1 Cc1ncsc1C(=O)N(CC(C)O)C1CC1.C(CCCN)N(C)C=O c1(C(=O)OCC)cocc1C(=O)NCCC1CC(NC(=O)CC2OCCC2C)C1 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC2CCN(C(C(C)C(F)(F)F)=O)C2C1 C1(C(=O)NCC2CCN2C(=O)CSCc2ccc(Cl)cc2)CC2CC1CC2(F)F C(CCCCC(=O)NC(CC1CCCC1)C(=O)NC(C)CCOC)OCC C1(C(c2c(C3(C)NC(=O)NC3=O)cccc2)NC2CCCC2)CC2CCC1CC2O N1(C(C(c2c(C)noc2C)C)=O)CCCN(C(=O)COC2CC2)CC1CO c1(NC(CN(CCOC)C(c2cccn2C)=O)C)cc(C#N)c([N+](=O)[O-])cc1C c1(C(=O)NC(CNC(C2(C(=O)OC)CCCC2)=O)(C)C)ccn2c(C)ncc2c1 C(c1ccc(CC)o1)=CC(=O)NCCC(C)N(C(C(CC)OCC)=O)C C(C(O)CC(=O)N(CC(C)(CC)OC)C)NC(c1c(CCC)n[nH]c1)=O C1(C(N(CCCNC(CNC(N)=O)=O)CCO)=O)CCCCN1S(N)(=O)=O c1(C(N2CCC(O)(c3cccc(F)c3)C2)C(=O)NC)cccc(OC(F)F)c1 N1(C(CC2(C=C)CC2)=O)CCC2(C1)CN(C(=O)CC(CC(C)C)n1ccnc1)C2 C1(NC(C2(O)CCOC2)=O)CCN(C(=O)COc2ccc(F)c(Cl)c2)C12CCC2 c1(OCC)ccc(C(=O)NCCC2(O)CCCN(C(=O)C(Cl)=CCl)C2)cc1OC C1(C(N2CCC(O)C2)=O)CCNCC12CC2 C1(NC(=O)C(C2CCCCC2)O)CC2CC1N(C(=O)CN1CCCNS1(=O)=O)C2 O=S(=O)(c1ccc(CNC2CCSCC2)c(F)c1)NCC1(C2=CCOCC2)CC1 Cc1ncccc1C(=O)NC(C)C(C)(C)NC(c1sc(F)cc1C)=O C1(CCN(C(c2cc(C)ns2)=O)C)CCCCN1C(=O)CC(O)C1CCCC1 CCCCCC(O)C(=O)NC(CC)CCCC(=O)N(C)Cc1occc1C C1(C(=O)NCC2CC(NC(C3CC(O)C3)=O)C2)CCC=CCCC1 C(C(CC)CC(C)C)NC(C(Cc1ccccc1Br)NC(C=CC)=O)=O N1(c2c(C)c(NC(C)CSCC(F)(F)F)ncn2)CCc2[nH]ccc2C1 c1(C(=O)NCC(CNC(CN2C(C)CC2)=O)O)cccc2c1oc1ccccc21 Cc1noc2ncnc(N3CCCC(CNC(=O)CSc4nncn4C)CC3)c12 c1(CC)nc2sc(C)cn2c1C(=O)NCC(C1CCCC1)NC(C1(O)CCC1)=O c1(OC)cccc(C(N2CCC(CC(=O)NCCCN3CCOCC3)C2)=O)c1F c1(CC)ccc(C(=O)NCCC2C(C)CCCN2C(c2n[nH]cc2C)=O)cc1Cl CCC(CC)C(C(=O)N1CC(CNC(C2CC(C(F)(F)F)C2)=O)CCC1C)OC C1(C(=O)NC(CCN(C(C2CC(OC)C2)=O)C)C)CC=CCC1C C(=O)(CCS(=O)(=O)NC)NC1CCC(F)(CNC(C(CC)SC)=O)C1 C1(COC)CN(C(=O)COCC2CC2(F)F)CCN1C(=O)COC1CCOCC1 c1(C(N(CCNC(c2ncc(OCC)nc2)=O)CC)=O)c(O)ncc2c1CCC2 C(C)(C)(CC(=O)N1CC2CC1C2CNC(c1ccc(Br)o1)=O)N(C)C C1(OCC=C)CCN(C(C2(n3cc(CCCOCCC)nn3)CCOCC2)=O)CC1 N1(C(c2c(C)cnnc2)=O)CC=C(C(=O)NCC(C)(C)OCCN(C)C)CC1 c1(C(=O)NCC(CNC(Cc2cn(CC)nn2)=O)O)ccc(C(F)F)c(OC)c1 C1(CN=C(NCCSC)N2CCC(c3ccccc3)C2)COc2ccccc2O1 Cn1nc2c(c1C(=O)NCC1CC1NC(=O)NC(=O)NCc1ccco1)CCCC2 CC(C)C(CCN(C)C(C1CSCCS1)=O)N=c1[nH]c(Cl)ncc1Cl Cc1cc(C(N2CCC3(CC2)CC3NC(c2cc(O)n[nH]2)=O)=O)ncc1[N+](=O)[O-] c1(NC(C(CNC(c2nnn(CC)c2C)=O)OC)=O)cn(C)nc1C#N Cc1c(C(=O)Nc2cccc(NC(=O)CC3CCC(O)C3)c2)nnn1C C1(CNC(c2ncncc2Cl)=O)CCC(F)(CNC(C2(C#N)CCCO2)=O)CC1 c1(C(=O)NC(CN(C)C(C2CC23CCC3)=O)(C)C)cc(=O)c2ccc(Cl)cc2o1 N1(C(Cc2ccc(C)cc2)=O)CC(NC(C2(C)CCCN2C)=O)CC1(C)C c1(NC(C2N(Cc3c(OC)cco3)C3C(C2)C3)=O)cc(O)ccc1[N+](=O)[O-] c1(C(N(CCNC(c2cc(C(C)C)[nH]n2)=O)CC)=O)nccc2ccn(C)c12 N1(CC(N2CC(CNC(C=COCC)=O)OCCC2)=O)C(=O)NC(C)(CC)C1=O c1(C(C(=O)N)n2cccc2)cc(F)cc(F)c1.C1(Cc2n[nH]cc2Br)CC(O)CN1 N1(C(C(C(C)(C)C)=O)=O)CC2CCCCC2(NC(=O)CC2=NNC(=O)C2)C1 N1(C(C2(C=C)CCC2)=O)CCN(C(=O)CC(C)C)CC2CCCCC12 N1(c2ccnc(NCc3nn(C)c(O)c3)n2)CCC2(CCC2)C(CO)C1 C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)C)NC(c1c(OC)scc1)=O c1(C(N(CCCOCCNC(C2CC(SC)C2)=O)C)=O)cnc(C2CC2)cc1C CC1CC(C(=O)NC(C)(C)CCNC(c2cc3[nH]ccc3s2)=O)CCN1C N1(C(CC)=O)CCC(C2CCCN2C(=O)CNC(=O)CNC(C)=O)CC1 C1(F)(CNC(c2nc(C(C)C)oc2)=O)CCN(C(C2CCCS2)=O)C1 C1(CNC(C(CC)n2ccnc2)=O)CCN(C(c2cn(CCO)nn2)=O)CC1C C(CC(C)(C)S(C)(=O)=O)CC(=O)N(CCCN(C)C1CC1)CC(F)F c1(C(N2CC(CCC)N(C(=O)CCNC(N)=O)CC2)=O)cc(C)c2[nH]cnc2c1 CS(=O)(=O)C1CCN(c2nnnn2-c2cnc(OC(=O)NC3CCC3)cn2)C1 C1(OCCn2cc(-c3c(C)ccs3)nn2)CCN(C(=O)Cc2cn[nH]c2)CC1 C1(C(N(CCCN(C(C=CC(=O)OC)=O)C)C)=O)CC1(C)C(C)C c1(C(C)=O)ccc2cc(C(N3CC(NC(C4CCCC4)=O)C4(CC4)C3)=O)[nH]c2c1 CC1CC(N=c2[nH]n(C)c(C(F)(F)F)c2[N+](=O)[O-])CN1C(C1C=CCCC1)=O c1(OCC(=O)NC2CC(CS(C)(=O)=O)C2)ccc(Br)cc1C#N S(=O)(=O)(c1[nH]c(=NC(C)CCC2CCCC2)ccc1Br)N1CCC(C(C)O)CC1 c1(C(=O)N(C2(C)CC(F)C2)C2CC2)ccc(Br)cc1 Cc1nc(C(=O)NCC2CCC(NC(c3cccc(Cl)c3)=O)CC2)nn1C c1(C(=O)OCCCCCC=C)cc(C(=O)OC(C)(C)C)cc(Br)c1C Cc1sncc1C(=O)NC(CO)C(C)NC(C1CC1C(N)=O)=O C1(C(=O)NC2(C)CN(C(CCc3ccn(C)c3)=O)C2)CCn2cnnc2C1 C12(CC)CC1CN(C(C1C(C)OCCN1C(c1ccon1)=O)=O)C2 Cn1ncc2c1CCC(C(N1CC3CC(Nc4cc(O)ncn4)C3C1)=O)C2 C1(CNC(c2cccc(C)c2)=O)C(C2CC2)CCN1C(=O)Cc1ccnn1C CC1(C)OCCC1CC(N1CCC2CC12C(=O)NCC1CCS(=O)(=O)C1)=O CCCCC(O)CC(=O)N1CCC(OCCNC(c2cccc(F)c2OC)=O)C1 N1(C(c2c(C(=O)OCC)ccs2)=O)CCCC2C1CCCN2C(C1CN(C)C1)=O c1(C(F)(F)F)cc2[nH]ccc2cc1-c1nc(C(F)(F)F)no1 Cc1nsc(C)c1C(=O)NCCC(C)N(C)C(c1cc(C(C)(F)F)n[nH]1)=O Cc1ccc(CCC(=O)NC2CCCN2CC(=O)NC(=O)NCC(C)C)s1 C=CCC(CC)C(=O)NC1(CO)CN(C(c2cnc(CO)nc2C)=O)C1 C=Cn1nncc1C(=O)N(C(C)C(N1CCCC1COC)=O)C1CC1 C#CC1(O)CCN(C(C2CN(C(c3ccc(C)n3C)=O)CC2CCC)=O)C1 Cc1nc(C(C)(C)C)c(C(=O)NCC2CCC2NC(=O)C=Cc2c[nH]nc2C)s1 c1(N(C2CCCN(C(=O)C(c3ccc(F)cc3)F)C2)C)ncccc1[N+](=O)[O-] C1(C(=O)NC(CNC(C(C)=CC2CC2)=O)C)CNc2ccnn2C1 N1(C(CNC=O)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1C1CC1 N1(C(C(CC(C)C)OC)=O)CC2CCCC(C1)N2C(=O)Cn1c(C)c(C)sc1=O C1(CC(=O)NC(C2CCN(C(=O)C(C)=C(C)C)C2)C)(CC=C)CCCC1 N1(C(c2ncc(CC)nc2)=O)CCC(O)CC1C(N1CC2CC1CS2)=O Cc1cc(CNC(=O)C(CCC2CC2)NC(c2nocc2C)=O)cc(C)n1 C1(CC)(NC(=O)C(C)SC)CCCN(C(c2ccc(Cl)cc2OC)=O)C1 C12(NC(C(COC)NC(=O)CCc3cn(C)nn3)=O)CC1COC21CCC1 c1(NCC)cccc(F)c1C(N1CCN(C(=O)COC2CC=CC2)C(C)C1)=O c1(C(=O)NCC(CNC(C(C(C)C)SCC)=O)O)ccc(O)cc1[N+](=O)[O-] N1(C(c2cccc(C)n2)=O)CC2CCN(C(C34CC3COC4(C)C)=O)CCC2C1 N1(C(C(CC(=O)OCC)C)=O)CCCC2(C1)CN(C(=O)CCC(C)C)C2 N1(C(c2nc(OC)sc2C(=O)NC2CCCCC2)=O)CC(NC(C)=O)CC(O)C1 c1(NC(C2N(Cc3ccc(CC)cc3)CC=C2)=O)cnc(C#N)c(C)n1 C12(C(=O)NC3C(CNC(C4CCOC4)=O)CCCC3)CCC(CC1)CO2 N1(C(Cc2c3cc(C)sc3sc2)=O)CCC2(CC1)CN(C(=O)Cc1cnoc1)C2 c1(C(N2CCCCC2CCNC(C2(C3CCCO3)CC2)=O)=O)[nH]cc2c1CCC2 c1(C(=O)C(N2CCC(c3cn(CCCCCO)nn3)CC2)=O)ccc(F)cc1F C(=O)(CCC(F)(F)F)NCCC(C)N(C)C(c1ccc(CO)nc1)=O C(=O)(C1=NOC(C(N2CC3CC2C3CNC(=O)CC2CC2(C)C)=O)C1)OC C(C(C(=O)N1CC(c2cc[nH]n2)C1)C(C)(C)C)NC(C1N(CCC)CCC1)=O C1(C(CNC(c2c(NC(C)=O)ccs2)=O)=O)CSc2ccccc2O1 C12(C(=O)NC(C)CNC(=O)C(=O)N=S(C)(C)=O)CCC(N=[N+]=[N-])(CC1)C2 C1(C2(O)CCN(C(=O)C(C)(F)CC)CC2)(NC(C(CC)n2nccc2C)=O)CC1 C1(C(=O)Nc2c(C)nsc2)CCCN(C(C2(C)CC(C)(C)C2)=O)CC1 C1(OCC)CCCC1NC(=O)C=CCNC(=O)CC1CCOC1C C1(CNC(c2ccc(CCC)[nH]2)=O)COCCN(C(c2c(N)cccc2Cl)=O)C1 N(C1COCc2ccccc21)C(C1CCC(NCc2cc(I)ccc2F)C1)=O c1(OC)ccc(CCC(N2CCCCC2CN(C)C(C2CC2C)=O)=O)cc1Cl c1(CC)ccc(C(=O)NC(C)(C)CNC(=O)CCC2CC2(Cl)Cl)c(C)n1 C(C)(c1ccsc1)=CC(=O)NCC(C1(O)CN(C(C2C(CCC)C2)=O)C1)(C)C c1(COC(=O)CC2(C(=O)OCC)CCCC2)cc(Cl)c(Cl)cc1Br C12(C(=O)NC3C(NC(C(C)OCC=C)=O)CCC3)CC3CC(C1)CC(C)(C3)C2 c1(OCCOC)cccc(-c2cn(C(C)(C)CC(=O)NCC3CC(O)C3)nn2)c1 CCC(CCCC(=O)N1CCC(N(C)C)C1C)NC(C1CC12CCCC2)=O c1(C(=O)NCCC2CCN(Cc3cccc(OC)c3)C2)ccc2c(c1)CCO2 C1(C(=O)NCC2(C(N(CCC#C)CC)=O)CCC2)CC2CC(=O)C1O2 C=CC(C)(C)CCNC(=O)C(CC=CC)NC(c1sc(C)nc1C)=O C1(C(=O)NCCCC(C)CO)CCN(C(c2cccc(=O)n2C)=O)CC1O C1(CCCC)(C(=O)N(C2CC(N(C)C)C2)C)CCCCC1.C12(CC1)C(=O)NC2 c1(SCC)ccc(C(N2CCN(C(c3conc3C)=O)CC2)=O)cn1 N1(C(c2scc(C)c2)=O)CCCC(NC(c2ccc(N)nc2)=O)CC1 C(=O)(C(CC(N)=O)NC(=O)CN1CCCC1C)NC1(CCC)CCOC1 CC1(C)CC(C(=O)NC2(CCNC(C3CC4COCC4C3)=O)CCC2)CCO1 CC(C)CCCCCN(C(=O)CNS(=O)(=O)c1cccs1)C(C)C Cc1nc(NCCCCCCC2CC2)cc(=NCC2CCCC(F)C2)[nH]1 C(=O)(C(C)(C)C(F)(F)F)NC1CCCC(NC(C(CC)(C)F)=O)C1 c1(C(N2CC(OCCNC(C3C(C)(CC)C3)=O)C2)=O)cc2n(n1)CCC2 C(=O)(C1=CC(C)(C)C1)N(C(C(=O)NC(C)C)C1CC1)C N1(C(c2n(CC#C)ccc2)=O)CCCC(C)(C(=O)NCC2CCCS2)C1 c1(C(=O)NCC(C(C)(C)C)NC(C2ON=C(CC)C2)=O)cc(C#N)cn1C N1(C(C2N(C(N)=O)CCCC2)=O)CCC(NC(=O)CCC2CC2(Cl)Cl)CC(O)C1 c1(OCC)ccnc(CCC(N2CCCC2c2cn(CC3CC3)nn2)=O)n1.OCC C1(C)(C(N(C(CC#C)C)C)=O)CC(NC(=O)C(C)CC2CCCC2)C1 c1(C(=O)NCC2N(C(c3cc(C)on3)=O)CCCC2C)nccc2ncccc12 C1(C(N2C(CN(C)C(C3Cc4nncn4C3)=O)CCC2)=O)CCC12CCOCC2 c1(C2C(C(=O)NCC3N(C(C(C)=C(C)C)=O)CC3)C2)nnc(S)n1C N(C(=NCC(C)C)NCc1cnc(C)s1)C(c1ccc(OC)cc1)C N1(CCc2c(C)nn(C)c2)CCC(=O)N(CC2(C(F)(F)F)CC2)C1=O c1(NCCCC=C)ccc(S(=O)(=O)NCC2CCN(C(=O)CC)C2)c(Br)c1 C1(NC(=O)CC2CCCC2)CCN(C(c2cc[nH]c2)=O)CC1F c1(-c2nc(N3C(C)CCC(c4c(C)coc4)C3)on2)ccc(S(=O)CC#N)cc1 C1(CNC(C2(F)C(C)C2)=O)CCCN1C(c1cc(CS)cs1)=O.C(C)(C)(C)O N1(C(Cc2n(C)ccn2)=O)CCC(C)(CNC(=O)CCN2CCCC2=O)CC1 C1(NC(=O)Nc2ncccc2Cl)CN(CC(N2CCCC2)=O)CCC1(F)F N1(Cc2n(C)ncc2)CC2CCC1CN2CC1(c2ccccc2)CCCCO1 CC(C)C(C)CC(=O)NCC1(O)CCCN(C(=O)Cn2ncn(C)c2=O)C1 N=c1[nH]cc(C(=O)NOC2(C(=O)O)CC2)s1 C1(NC(C2CN(C(C)C)C2)=O)CC2(CCCCN2C(=O)CCc2nncs2)C1 c1(C(=O)NCCN(C(C(C)S(C)(=O)=O)=O)CC2CC2)ccc2c(c1)COCC2 N1(CC)CCN(C(c2ccc(F)cc2OC)C(=O)NC2(C)CC2)C(C)C1 O=C1CCN(CC2CNC(=O)C2(F)F)C(=O)N1CC1=CCCOC1 C(=O)(C(O)C1=CCCCC1)C(N1CCCCC1Cc1cn(CCCCO)nn1)=O C12(NC(C(C)NC(N)=O)=O)CCCC1N(C(c1cccc(F)c1N)=O)CCC2 c1(C(=O)NC(C2CCCN(C(c3cn(C)nc3O)=O)C2)C)cc(F)cc(Br)c1 C1(NCc2ccn(C(C)C)n2)CCCC2NCCC12 c1(OC)ccc(C(C2CCNCC2)NC(=O)Cc2csc(C#N)c2)cc1F C1(C(=O)NC2C(OC)C(C)(C)C2)CC(C)CN(C(=O)CC2(O)CCCC2)C1 N1(C(CCC=C)=O)CCCC2(CC(NC(C3Cc4ccncc4CO3)=O)C2)C1 C1(OC)CC2CCC1CC2C(N1CCC(NC(=O)CC2CS(=O)(=O)C2)C1)=O c1(C(N2CC(C)CC(NC(C=C(C)C(F)F)=O)C2)=O)cc(S(N)(=O)=O)ccc1C c1(OC)cccc(C(=O)NCCCC2CCN(C(C3CC3(C)C)=O)CC2)c1Cl c1(N2C3C(N4C5CN(C(C)=O)CC54)C(C3)C2)nc2c(C)cccc2o1 C(C)(CCCC(=O)NCCC1CC1)NC(Cc1cc(C)[nH]n1)=O C1(F)(C(=O)NC(C(=O)NC)CC2CC2)CCN(C(=O)CCc2cnn[nH]2)C1 C(=O)(CC(C)C(=O)N1CCC(C=CC(=O)Nc2cc(OC)cc(O)c2)CC1)OC Cc1noc(C(=O)NCC(O)CCNC(C2CC(N(C)C)C2)=O)n1 C1(C(N(CC#C)CCOC)=O)CCC(C2CC2)N1C(=O)Cn1ccnn1 N1(C(Cc2ncc(C)o2)=O)CC(NC(c2ccc(F)c(F)c2)=O)CC(O)C1 N1(C(C=C(C)C(F)F)=O)CCC(NC(c2ccc(CS(C)(=O)=O)o2)=O)C(C)(C)C1 C1(CNC(COCc2cccc(C)c2)=O)C(O)C(O)CN1C(=O)C(C)C#N C1(NC(c2sc(C)c(Br)c2)=O)CC2CC1N(C(c1csnn1)=O)C2 c1(C(=O)NCC(C)NC(C2(CC)CC2)=O)cc(SC)oc1C CCC(CC(=O)NCC1C2CC1N(C(c1sc(C(C)C)nc1C)=O)C2)C(C)C c1(CN(C(C(C(C)C)CN(C)C)=O)C)cn2c(n1)CCCC2 C1(CNC(C(C)NCc2ncc(C)c(Br)c2)=O)CCCCC1C1CC1 C1(CN2C(=O)CCN(CC34CCCC3C4)C2=O)CCCS(=O)(=O)CC1 C1(C(=O)NC2CN(C(C34CC(CC(F)F)(C3)C4)=O)C2)CCCCC1 c1(OC)ccc(CN2CCCC(CNC(=O)CC3CCCOC3)C2)c(OC)c1 C(=O)(C#CC1(C)CCCO1)NC12C(CN(C(C(C)OCC=C)=O)C1)CCC2 n1(CC)cc(C(N2CC3CC3(CNC(C3CCNC3=O)=O)C2)=O)c(C(F)(F)F)n1 C(=O)(C(CCCC(C)(F)F)NC(=O)OCC(C)(C)C)Nc1c(C)c(C#N)ccc1 N1(C(Cc2cc(CC)no2)=O)CCC(C)(C)C1C(=O)NC1CCC(N(C)C)C1 C(=O)(CC(CC)C(C)C)N(CC(C)(C)C(=O)NCC(C)(C)CNC(=O)C(C)C)CC C1(NC(C(CC)=CC)=O)CCC2(CC1)CC2NC(=O)C(=O)NCC N1(C(C(C)C(C)(C)C)=O)CC2CCN(C(=O)C(C)(C)CO)CCC2C1 c1(C(N2CCC(C)(CNC(=O)CC3COCCOC3)C2)=O)cccn2nccc12 c1(C(N(C2CCN(C(C3=C(C)OCCS3)=O)C2)C)=O)cc2c(cc1Cl)NC(=O)C2 N1(C(C(=O)NC2CCCN(c3ccccn3)C2)=O)CC2CCNCC12 C(=O)(C1CCNc2cc(F)ccc21)NC(C1CN(C(C2CC(C)(F)C2)=O)C1)C Cc1cccc(C(F)(F)C(=O)NCC2CCN2C(C2CCCC23CC3)=O)c1 C1(NC(C(C)Cc2ccccc2Cl)=O)CN(C(=O)Cc2cn[nH]c2)C(C)(C)C1 c1(C(N2CC(NC(=O)COCC3(F)CC3)C(O)C2)=O)ccc2nnn(O)c2c1 N1(C(C2(COC)CCCCC2)=O)CCCCC2(CCN(C(=O)C(C)C(C)O)C2)C1 N1(CCC)CCCC(C(=O)NC2CCC(CNC(c3cccnn3)=O)C2)C1 C1(C(N2CCC(N(C(=O)COCC3CCCO3)CCC)C2)=O)NC(=O)OC1(C)C C1(NC(CCC(C)OC)=O)CCCC2CN(C(=O)C(C)Cc3cnn(C)c3)CC12 c1(C(=O)NCC(C(C)C)NC(C2(C)CCCO2)=O)cc[n+]([O-])cc1 Cn1ncc2c(O)nc(NC3CC(CNC(c4csc(C(F)F)n4)=O)C3)nc12 c1(OCCNC(CC(COC)C)=O)ccc(C)cc1C.C1CO1 N1(C(CCC(C)OC)=O)CCOCCC1C(=O)NCCOc1cnn(C)c1 CC12CCN(C(c3nccs3)=O)C1CN(C(C1CCCC3(C1)CC3(F)F)=O)C2 c1(C(N2CC=CC(NC(C3CCC34CCC4)=O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] C1(C(C)C)CN(C(c2coc(N3CCOCC3)n2)=O)CCN1C(C1CC12CC2)=O N(C(=NCCCc1nnc(C)n1C)NC(C)COC)C(CC)C(F)F C1(CNC(C2C(C=C)C2)=O)CN(C(c2csc(S)n2)=O)CCCO1 C1(C(N2CCCC(OC)C2)=O)C2CCCC1CN(C(c1cc(Cl)nc(Cl)c1)=O)C2 C(=O)(CCC(C)(C)C)NCc1ccc(C(N2CCCC(OC)C2)=O)o1 c1(C(N(C(C)C)CCc2nn[nH]n2)=O)n[nH]c(C2CCCO2)n1 c1(SCC(=O)NC(CN(C(=O)Cn2ccnn2)C)(C)C)n[nH]c(O)n1 c1(NCC)ccc(F)cc1C(=O)NC1CC1NC(=O)CC(C)CN(C)C C(CCCCCN=c1ccc(S(C)(=O)=O)c[nH]1)NC(C(CC)NC(C)=O)=O c1(C(N2CCC(C)C(CNC(c3c(Cl)nsc3Cl)=O)C2)=O)cnc(O)n(C)c1=O C#Cc1cc(F)c(COC(C23CCN(C(=O)OC(C)(C)C)CCCC2C3)=O)c(F)c1 N1(C(C(CC)N(C)C)=O)CC2(COC(CNC(=O)C(F)=CC3CC3)C2)C1 C(=O)(CN1C(=O)CCc2ccccc21)N1CCC(NC(CC=C)=O)CC1C c1(C(N2CCC(C(=O)Nc3cc(F)c(F)cc3Cl)C2)=O)cc(O)cc([N+](=O)[O-])c1 CC1=C(C(=O)NCC2C(C)CCCN2C(c2nnc3n2CCCC3)=O)CCCO1 c1(OC)cccc(C(=O)NCCN(C(=O)C(C)(C)CC2CC2)C2CC2)c1 C(=O)(C1=CCCCCC1)NC1CCN(C(Cc2c(OC)ccc(F)c2)=O)CC1O N1(C(C(C2CC2)NC(c2nc(C)oc2C)=O)=O)CCC2CN(C)CCC12 c1(C(C(C)NC(CNC(=O)OC)=O)NC(=O)CCNS(C)(=O)=O)ccccc1 C1(C(C)NC(C2CCC2)=O)CCN(C(=O)C=C(Cl)Cl)C1 C1(NC(=O)CC2(CO)CCC2)CC(O)CN(C(=O)Cc2ccon2)C1 N1(C=O)CC(NC(=O)OC(C)(C)C)C2(CC2)C1.C1(CCOCC)(OC)CC2CCC1C2 N1(C(C2CCC(C(N)=O)C2)=O)CC(CO)CC1(C)C.CC1(C)C2C1C(=O)N2 CC(C)C(C(=O)NCC1(CCNC(C2CC(Cl)(Cl)C2)=O)CC1)n1cncn1 c1(NC(=O)NC(c2c(C)[nH]c(C(=O)NCCCl)c2C)=O)c(Br)cc(Br)c(C)c1Br C1(C(N2CCC(SC)C2)=O)(NC(C=CC(CC)C)=O)CCN(C)C1 c1(CC)nc(C)c(CN2CCC(COC3CCN(C)CC3)C2)[nH]1 CCCCCCC(=O)N1CC(CC)C(CCNC(=O)C(F)(F)CC)C1 N1(C(C2CC(SC)C2)=O)C2CC1CN(Cc1ccc(C)c(C)n1)C2 N1(C(c2c(CC)con2)=O)CCCC(C)C1CNC(=O)CCCCc1cnn[nH]1 C1(CNC(CC2CC(OC)C2)=O)CN(C(=O)C=CC2CCOC2)CC1S(C)(=O)=O c1(NC(c2cnc(-c3ccc(C(=O)O)cc3)nc2)=O)cc(F)cc(Br)c1Cl CC1CC2CN(C(=O)CN3CCCC3CO)CC2N1C(c1ccc([N+](=O)[O-])[nH]1)=O c1(C(=O)NC2CCC(CCNC(c3c(C)nn[nH]3)=O)C2)c(Cl)csc1Cl N1(C(Cn2c(C)csc2=O)=O)CCCC2C(CCCN2C(=O)CN(C)CCO)C1 c1(C(=O)NC)cccc(C(=O)NCCCNC(=O)CN(C)CCO)n1 C=CC(CCC)CC(=O)N1CCC(CN(C(=O)Cc2[nH]cnc2C)C)C1 CC(C)C(C)CC(=O)N(C1CCC(NC(=O)COC2CCOC2=O)CC1)C N1(C(CC2N(C(C)=O)CCC2)=O)CCCCC1CNC(=O)CC1OCCC1(C)C N1(C(=O)CCNCCCO)C2CN(C(c3cnc(Cl)nc3)=O)CC12 CN1CCC(NC(=O)Cc2cccs2)C12CCCN(C(=O)C(F)C1CCOC1)C2 C1(CNC(CCNC(=O)CO)=O)CC2CN(C(c3nc(C4CC4)cs3)=O)CC12 N1(C(C2(CNC(C3C(OCC)CC3)=O)CCOC2)=O)CCC(C)(CO)C1 CC1(NC(C2CC2F)=O)CCN(C(c2ccc(C(F)(F)F)o2)=O)C1 C1(CNC(c2[nH]c(=NC)sc2)=O)CCN(C(c2ccc(Cl)nn2)=O)CC1C N1(C(C(C)=O)=O)CCOCC2(COCCN2C(=O)C#CC2CCOC2)C1 c1(NC(C2C(SCC)CCCC2)=O)nn(C)c2c1CS(=O)(=O)CC2 C1(CNC(C(=O)NC(C)C)=O)(CO)CCN(C(C2CC23CCCC3)=O)CC1 CC(CC(=O)N1CC(CNC(c2cccnc2-n2cncn2)=O)C1)C(F)F N1(C(C2C(COC)CC2)=O)C2CCC1CC(CNC(C1(C#N)CC1)=O)C2 c1(CC(=O)NCC(C(C)(C)C)NC(=O)C(F)=CC2CC2)c[nH]c2ccc(Cl)cc12 CC1(O)CCN(c2ccc(-c3c(CO)cccc3)cc2Br)CC1O C1(C(=O)NCCCC)CC(C)CCN1Cc1nc(O)n[nH]1 C1(C#N)(C(=O)NC2CC(CC(=O)NCc3ccn(C)n3)C2)CCCC1 C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1N(C(C2CC23CCSCC3)=O)CCCC1 C(=O)(CCCC(=O)N(C)C)NC1CC(F)(CNC(c2c(C)nncc2)=O)C1 n1(CC)nc(C(C)C)cc1C(=O)NCC(C)(C(C)C)NC(=O)CCc1cccs1 c1(C(=O)NCCC2(n3cc(Br)cn3)CC2)cccc2c(I)n[nH]c12 CCC(C)(C)C(=O)C(=O)N1CC=CC(NC(c2csc3nnsc23)=O)C1 N1(C(C2(C=C)CC2)=O)C2CCC1(CNC(=O)CC(C)(C)c1ccc(F)cc1)CC2 N1(C(c2c(C)ncs2)=O)CC2CCC(NC(=O)CC3CC4(CCCC4)CO3)(C2)C1 C1(C(N2CCC(CN(C)C(c3ccc(OC)cn3)=O)C2)=O)CCc2nncn2C1 c1(C(N(C(C)CCNC(c2ccoc2Cl)=O)C)=O)cccc(C2CC2(F)F)c1 C(c1cc(Cl)cc(Cl)c1)=CC(=O)NC1CCN(C(c2cnc(OC)s2)=O)CC1 C1(C)(CNc2ccc(OCC)cc2)CCCN(C(=O)CC2CCOCC2)C1 C(=O)(C(C)C1=CCCC1)NCC(CC)NC(=O)Cc1ccc(OC(F)F)cc1 Cn1nccc1CC1(C(=O)NCCCCNC(c2sccc2Cl)=O)CC1 c1(C(=O)NCC2(C)CN(C(=O)C=CC3CC3)CCO2)nnc(O)c(Br)c1O C1(C(C(=O)NC2CN(C(C=C(COC)C)=O)C2)C)CCOCC1 C1(C(=O)Nc2scc(-c3cn(C(CC)C)nc3)n2)COCCN1C(=O)COC c1(C(=O)NC(C2CCCC2)CNC(C2CC(=C)C2)=O)cnc2n1CCC(C)C2 c1(OC)ccccc1-c1nc(CCCO)nn1Cc1ccc(I)cc1 CS(=O)(=O)c1cc(N2CCCC2CNC(=O)Cc2cccnc2)ncn1 N1(C(=O)NC(c2cccc(Cl)c2)C(F)(F)F)CCOC(c2ncno2)C1 O=C1NCC2(CCCN(C(=O)Nc3ccc4sccc4c3)CC2)C1O c1(CC(C)NC(c2cc(CNC(c3coc(CO)c3)=O)[nH]n2)=O)nncn1C N1(C(C(C2CCN(c3nnnn3C)CC2)C)=O)CC2(CCC2)C1C1CCCO1 CC(CCCCN=c1ncc(F)c[nH]1)NC(=O)CCOCC1CCCO1 C(=O)(CC(C)C(=O)O)N(c1ncc(-c2cn(CC(C)(C)C)nn2)n1C)C Cc1cc(F)sc1C(=O)N(C)CCN(C)C(c1cccc(-c2nnco2)c1)=O C(=O)(CCCC(F)(F)F)N1CCC(NC(c2nccc3cc[nH]c23)=O)CC1 O=C(CC(C(F)(F)F)NC(=O)Cc1cccnc1)NC(CCO)C1CCCC1 c1(C(=O)NCC2(O)CCCN(C(=O)CCC[N+](=O)[O-])C2)ccc2c(c1)CCO2 c1(CC)nc(C)c(CC(=O)NCCC(C)(C)NC(C2(C)CCCC2O)=O)c(C)n1 C=C(C)CC(C(=O)NCCCN(CC)CC)NC(=O)Cc1cncc(C)c1 C1(OC)CC(NC(C2CC3C=CC2O3)=O)CN(C(=O)CN2CCC(CO)CC2)C1 C1(NC(c2ccc(C(N)=O)cn2)=O)CC2CC(NC(c3sccc3CO)=O)C1C2 C1(CC(=O)NCCCOCCNC(C2(OCC)CCC2)=O)CC(=O)N(CC)C1 C1(C(N2C(CNC(c3c(C)cns3)=O)CC2)=O)CCC(O)CN1C C1(CC)CCC(O)(C(=O)NCc2nc(CNC(c3sccc3C(C)C)=O)cs2)C1 c1(OC)ccc(C(=O)NC(C2CCCN2C(c2ncncc2Cl)=O)(C)C)cn1 CC(C)(C)C1=NOC(CNC(=O)C(N2CC3CCC2C(O)C3)=O)C1 c1(C(N(CCN(C(=O)CC(C)C2CCCO2)CC)CC)=O)ccnc(O)c1F C1(F)(CNC(c2c(C)ccnn2)=O)CCC(CNC(C2CCNC(=O)C2)=O)CC1 N(C(=NCCNC(=O)NC1CCCC1NCC)NSC)C(CC)C.C(C(F)(F)F)O C12(NC(CSCC(N)=O)=O)CCC1CN(C(=O)CCc1cnc(C(C)(C)C)o1)C2 N1(CC(=O)NC(CC)C)CCCc2cccc(Br)c21.c12cc(C)ccc1C(=O)O2 CCC(CCC(=O)NC1CC2CC1CC2C(=O)NCC1CCCC(OC)C1)OC c1(C(N(c2nnnn2CC(F)F)C)=O)ccc(Br)cc1C(F)(F)F Cc1nc(C(=O)NC2CN(C(=O)CCCc3ccsc3)CC2F)c(C)s1 N1(C(C2CCN(C)C2)=O)CCN(C(c2cnoc2-c2ccco2)=O)C2CCC12 C=C(CNC(=O)C(CC(C)C)N(C)C(C1CCCC(=O)N1)=O)C1CCOCC1 c1(C2C(CNC(c3cnc4c(Br)cccn34)=O)C2)cccc(C2=CCOC2)c1 C1(CC(=O)NCCOCCCNC(C2SCCCS2)=O)CCC2(CCC2)O1 CC1(C)CC(CC(=O)NCC(C)(CO)N2CCOCC2)N(C(C2OCCCO2)=O)C1 c1(OC)cc(C(=O)NC(C)CN(C(=O)CCC2(C)CCC(=O)N2)C)c(Cl)cn1 C1(C(N(C2CCN(CC)CC2)CC)=O)Cc2ccccc2C1.C(=O)(CSC)NCC C#Cc1cn(C)nc1C(=O)NC(CCN(C(=O)C(F)=CCC)C)C(C)C CC(C)(CCCNC(c1cccs1)=O)C(=O)N1CC2(CNC(=O)C2)C1 N1(C(C(C)Oc2cc(C)cc(C)c2)=O)CCCC12CCCN(C(=O)CCF)C2 c1(-c2cc(OC)cc(C#N)c2)ccc2c(c1)CN(C(C1(CF)CC1)=O)CC2 CN1CC(O)CCC1C(=O)NC1C2CC3C1C3C2C(=O)NCCOC(F)F c1(C(=O)NCC(C(=O)NCC(C)(C2CC2)OC)O)ccc(C)nn1 C(=O)(C(F)CC(C)C)NC(CC)CNC(C1(c2ccnn2C)CC1)=O C(=O)(C1CCCc2ccnn21)N1C(C)CCC(NC(=O)C2=NNC(=O)CC2)C1 CC1(C2CC(=O)NC2=O)CCN(C(C23CCCC2C3Br)=O)CC1 c1(C(=O)NC2(CNC(CC(=O)OC)=O)CCCCC2C)nc2cc(F)ccc2s1 Cc1cc(C(=O)NCC2=CCN(C(C3CCCC(F)C3)=O)CC2)cc(Cl)n1 C1(C#N)(C(=O)NCC2(O)CC(C(=O)NCCC(C)CCO)C2)CCCOC1 c1(C(N2CC3C(CNC(C(CO)NC(N)=O)=O)(C3)C2)=O)ccc(C(F)F)nc1O C(C(C(=O)NC(C)CCCC1CC1)C(C)C)NC(C(CC=C)OC)=O C1(CC=C)(C(=O)NCCCc2ncc[nH]2)CN(C(c2cn(CCOC)cn2)=O)C1 C1(C(=O)NC2CN(C(c3cc(C#N)on3)=O)CC2O)CCCCC12CCC2 Cn1ncc(NC(=O)OC(C)(C)C)c1S(=O)(=O)NOCc1ccc(Br)cc1 c1(N(CCN(C(C)C)C(C2CC3(C2)CC3F)=O)C)ccnc(S(C)(=O)=O)n1 C1(NC(c2nnn(C(C)(C)C)n2)=O)CC(NC(c2c[nH]ccc2=O)=O)C12CCC2 Cc1cc(C(N2CC3(CNC(C4CC(O)C4)=O)CCC2C3)=O)nc(O)c1 C(CC(=O)NC1CCCC(O)C1)(C(C)OC)NC(COCCOCC#C)=O C(N=c1[nH]c(=NC2CCN(C)C2)[nH]c2c1CSC2)c1nc(C)c(C)[nH]1 c1(Nc2nccc(=NCC3(COC)CCOC3)[nH]2)c(C)ccc2ncccc12 c1(OC)c(C(N2CC(C)C2C(=O)NCC2CN(C)CCO2)=O)cnn1C c1(CC)ccc(C(=O)NCc2occc2C(=O)N(CC(F)Cl)C)nc1 Nc1cnc(Cl)cc1C(N1CCC1CNC(=O)CC(O)C1CC1)=O C1(CC2(NC3C(C(=O)NC)C3C)CC2)CN(C(c2cccnc2)=O)CCC1(F)F C(C)(CO)(C(=O)N(CCCCCNC(=O)C(C)c1ncco1)C)OC c1(C2C(C(=O)NC3CCN(C(CCC=C)=O)CC3)C2)ccc(S(N)(=O)=O)cc1 C12(CCOCC1)C(=O)N2.c1(COC)cccc(C(=O)N(C(C)CS(C)=O)C)n1 c1(C(=O)NC2CCCN(C(C3(C=C)CCCCC3)=O)C2)cc(C)c(C#N)c(C)c1 N1(C(c2cc(Br)cnc2SC)=O)CCN(C(C(CCC)C)=O)C(CC)C1 c1(NC(C2CCCN(C(=O)CN3CCCCC3)C2)C)cc(C2CC2)ncn1 N1(C(C(=O)NCc2nnc(C)c(C)c2C#N)=O)CC2COC(C)(C)OCC2C1 CCC(CC(=O)NC(c1ccc(OC)cc1)CNC(C1CNC(=O)C1)=O)SC C(=O)(C(C)(C)CF)NCC(C)(F)CNC(C1CC1(Cl)Cl)=O C(=O)(CC(C)(C)C(C)(F)F)N1CC(C)N(C(c2nonc2N)=O)CC1 N1(C(C(CC=C)C)=O)CC2(C1)SCCC2NC(c1ncc(C)cc1OC)=O Cc1sc(Br)c(C(=O)NC(C)CCCNC(C2(O)CCOC2)=O)c1C N1(C(C)C(N2CCCC2CNC(C2SCCCS2)=O)=O)CCCCC1C N1(C(CCc2ccc(SC)cc2)=O)CCC(NC(=O)CC2CCC(=O)N2)C(F)C1 N1(C(C23CC(CCC)(C2)C3)=O)CC(NC(=O)CC23CCCC2C3)C2(CC2)C1 C1(C(=O)NCC2C(C(C)C)OCC2)C=CCCN1C(c1cc(=O)cc[nH]1)=O c1(OC)c(C(c2nnnn2C2CCC2)NC2C3CCCCCC23)cccc1F N1(C(C(COC)C)=O)CCCC1(C)CNC(c1ccc(CC#N)cc1)=O C(=O)(CCCCC(N)=O)NCCCC(C)NC(=O)C(C)NC(c1cncs1)=O N1(C(C(CCCC)F)=O)CC2(C=C(C(=O)NCc3oc(CC)nc3C)CO2)C1 N1(C(C(C(C)C)=O)=O)CCOCC(C(=O)NC(C)C(N)=O)C1 N1(C(C(C)OCC=C)=O)CCC(CN(C(=O)C(C)C2(O)CCC2)CC)C1 C1(NC(C2CCC(O)C2)=O)CCN(c2nnc(CO)s2)CCC1CO Cc1c(C(=O)NCC2CN(C(c3cc(OC(C)C)ccn3)=O)C2)cccc1C#N C(=O)(C(C)C(O)C(C)CC)N1CC=C(C(=O)NC(CC=C)CC(F)F)C1 c1(NC(N2CCC(c3nc[nH]n3)C2)=O)ccc(N2CCC2=O)cc1 c1(C(N2CC(CC(C)(C)C)N(C(=O)CSC(F)F)CC2)=O)ccn2cnnc2c1 C1(C(F)(F)F)(CN(C(=O)C(C)(C)OCC(F)(F)F)C)CCOCC1 c1(CC)ccccc1CCNC(c1ccc(-c2nncn2CC)cc1)=O Cc1nn(C)c(=O)c(C(=O)NC2CCCCC2Nc2ccnc3ncnn23)c1C N1(C(C(C)CF)=O)CC(NC(c2cc(C3CC3)nc(O)c2)=O)C(C2CC2)C1 N1(C(CC2CC(=C)C2)=O)CCCC(C2CN(C(c3cnc(C)cn3)=O)C2)C1 Cc1c(N2CCC(C)(CC(=O)O)C2)ncnc1Cl.C n1(CC(=O)NCC2CCN(C(c3nn(C)nc3Br)=O)C2)cnc([N+](=O)[O-])n1 C=CC(CCC)CC(=O)NCC1(C)CN(C(=O)C(=Cc2cccs2)C)CCO1 CCCCCC=CC(=O)NCC1CN(C(=O)C(C)(C)n2cc(Cl)cn2)C1 N(C(=NCC(C)C)NCc1ccnc(C(F)(F)F)c1)CC(CC)C(C)C C(=O)(CC(C)(C)C#N)NCC1C(NC(c2cccc(NS(C)(=O)=O)c2)=O)C1 C1(NC(C=C(COC)C)=O)CCCCC1CNC(=O)CCC1(C)CC1(F)F c1(NC(=O)OC(C)(C)C)ccc(N2CCN(Cc3scnc3Br)CC2)cc1 c1(C(=O)NCCOCCCNC(=O)COO)cc(O)nc(O)n1.C1(CN)CCCCO1 C1(C(=O)NCC(CC(=O)N(C2CCCC2C#N)C)OC)CN2CCN1CC2 C1(NC(c2nnc(O)cc2O)=O)CCN(C(=O)C(F)=CC2CC2)C12CCC2 c1(C(=O)NCCC(CNC(CS(CC)=O)=O)O)nc(-c2ccccc2)ncc1Cl c1(CC(C(=O)NCCCN(C(c2ccccc2O)=O)CC)C)c(C)noc1C c1(C(=O)NC2C(NC(c3cnc(C)o3)=O)C2)ccc(OCCF)cc1 c1(OC)ccc(-c2ccnnc2)cc1-c1csc(C#N)n1 Cc1cc(C(N2CCCCC2c2cn(-c3cccc(N)c3)nn2)=O)cc(Cl)c1 c1(C(=O)NC2(CNC(CCc3c[nH]c(=N)[nH]3)=O)CCC2)ccn2ccnc2n1 Cn1nnc2cc(C(N3CCN(C(=O)CCCC4CCC4)C(CCO)C3)=O)sc12 c1(NC2CN(C(C#C)=O)CC2O)ncc(C)c(C)n1 c1(C(CNC(C23CCCC2C3)=O)NC(c2csnn2)=O)ccc(F)cc1F C(=O)(CC(C)CC(C)C)NCC(C(C)C)NC(C(COCC)(C)C)=O c1(CNC(Cc2cc(C(=O)OC)on2)=O)ccc(OCC(N)=O)cc1 C1(NC(C(CC)n2cccn2)=O)CCCC1(C)NC(=O)Cn1nccn1 C1(CNC(c2cnc[nH]2)=O)(NC(c2cccc(Cl)c2O)=O)CC2CCC1CC2 CC(CO)(C(=O)NCC1CCCCO1)NC(C1CC(F)C(=O)N1)=O c1(C(CNC(c2cc(Cl)n(C)n2)=O)NC(CC(CC)C)=O)ccc(F)cc1F C1(CC(=O)N(CCN(C(=O)C(C)(C)Cl)C(C)C)C)CCC(O)C1 c1(C(C)C)cc(CC(=O)N(C(C)CCNC(c2ocnc2C2CCC2)=O)C)on1 c1(C(C(=O)NCCc2c(CNC(CCCC)=O)nco2)F)ccc(F)cc1 CCCCCC(C)(C)C(=O)NCC(O)CNC(=O)C(C)(O)CC(C)(C)C N1(C(c2nc(C(C)C)oc2)=O)CCCC2(CNC(=O)CCc3cnccn3)CC12 c1(C(N2CCC(CN(C)C(c3cc(F)cs3)=O)C2)=O)cnc2cccnn12 N1(C(C2C(OC)CC2)=O)CC2CC(C(N3CC(c4ncccn4)C3)=O)C(C2)C1.C1(C)CC1 C#CCCC(=O)NC(C)C(c1ccccc1)NC(C1(CC(C)C)COC1)=O C1(C(=O)NC2CC(C(=O)NCC3(C(C)C)CC3)CC2O)Cc2nccn2C1 C#CCCC(O)C(=O)N1CCN(C(C)CNC(=O)CCc2cn[nH]c2)CC1 C(=O)(C1=C(C)CCOC1)N1CC2CC(C(=O)NCc3c(CC)c[nH]n3)(C1)C2 C1(CC(N2CCCC(N(C(=O)C(C)(C)c3ncco3)C)C2)=O)CCC(C)(O)CC1 Cc1ccc(C(=O)NC2(C)CCN(C(=O)CC3CC4C=CC3C4)C2)c(O)c1 C12(NC(=O)CN(C3CCCC3)C)CCC(CC1)C2(C)C.C12CCCN1C2C c1(C(N(c2cc(OC)c(Cl)nc2)C)=O)ccc(C2=CCC(C)CC2)cc1 C=CCC(CNC(=O)Cc1ccn(C)n1)NC(c1ccn(C2CCCC2)n1)=O N1(C(C=C(C)c2ccco2)=O)CCC2CCN(C(=O)CC(=O)N(C)C)C2C1 C1(CNC(C(CC)CO)=O)CN(C(C2CN(C(C)=O)C2)=O)CCC1(C)C c1(C(=O)NC2(C)CCCN(C(c3cccc(F)c3Cl)=O)C2)c[nH]c2cccnc12 c1(C(=O)NC2C(C)CN(C(C3CCCC3P(C)(C)=O)=O)C2)cccc2c1COCC2 CC1CCOC1CC(=O)NCCCCC1CN(C(c2cnn(CC(F)F)n2)=O)C1 C1(NC(C2N(C(Cc3nc(=N)[nH][nH]3)=O)CC=C2)c2ccccc2)CCCN(O)C1=O N1(C(C=C(C)Cl)=O)CCN(C(=O)C=CCCCC)C2(CC2)C1.c1(C)ccccc1F Cc1ccccc1C=CC(N1CCC(C)C1CNC(c1cnc2n1CCS2)=O)=O C=CCN=C(NCc1ncc(Cl)s1)NCc1ccccc1CS(N)(=O)=O c1(C(N2CCCC(CNC(Cc3nc(C)sc3)=O)C2)=O)cc2c(cn1)CCCC2 c1(NC(CC2N(C(c3ncc(OC)nc3)=O)CCOC2)=O)nccc(Br)c1Cl c1(OC)cc(C(N2CCC(O)(CCNC(C3CC(C)(C)C3)=O)CC2)=O)ccc1C C(=O)(CC(C)(C)C(F)F)C(=O)CCCC1(C(N2CC(C)SCC2)=O)CCC1 Cc1[nH]c(=N)sc1C(N1CCC1C(=O)Nc1ccc(-n2cccn2)cc1)=O Cc1c(F)cc(C(=O)NC(C)CCNC(C2CC=CCC2)=O)c(F)c1N C(=O)(C(CC)C(C)O)NCCCCCCNC(C(F)=CCC)=O c1(CC(=O)NCC2C(CNC(c3n(C)ncc3Cl)=O)C2)cccc(C#N)c1 c1(C(=O)NCC23C(C)OC(CC2)C3)n[nH]c2c1CN(C(=O)C(F)C1CCC1)C2 Cn1cc(Cl)cc1C(=O)NC1CN(C(C2CCN(c3ccncc3)CC2)=O)C1 N1(C(C(CN(C(=O)CN2CCCC2C)CC)F)=O)CC2(C(CN)CCS2(=O)=O)C1 C(=O)(CCCCC(=O)NCC(C1CCCN1C(c1ccncc1F)=O)(C)C)NC C1(C(C)(C)CNC(c2ccc(CO)o2)=O)CCCCN1C(=O)C=C1CCC1 c1(C(=O)OC)ccnc(Cl)c1NC(C1(F)CCN(Cc2cc(C)cc(O)c2)C1)=O c1(CC)ccc(C(=O)NC(C(=O)N(C)Cc2ccn(C)c2)C2CC2)s1 c1(OC)ccc2c(=NCCC(C)F)[nH]c(=NC3COc4ccccc43)[nH]c2c1 C12(C(=O)NCC3C4N(C(C56CCCC5CCC6)=O)C(CC4)C3)CCCN(CC1)C2 c1(C(=O)NCCC2CCN(C(C(CC)=CC)=O)C2)sc(OC)nc1C C1(C(=O)NCC2CCN(c3ccncn3)CC2)CCN(C(=O)C2CC2)O1 C(C(CC(C)C)NC(=O)CCC1CCCOC1)NC(C1CC(C(C)C)C1)=O N1(C(C(C)N(C)C)=O)CCC(C)(C)C(NC(=O)CC2(n3cccn3)CC2)C1 CC1CN(C(=O)CN(C2CCC2)C(C2CC(=O)CC(=O)N2)=O)CC(=O)N1C CCCCC(CC)C(=O)NC1CCC(CNC(c2c(C)cccc2N)=O)C1 CC(C)(C)C(O)CCC(=O)N1CCN(C(c2cc(O)cc(O)c2)=O)CC(O)C1 N1(C(c2c(C(C)C)c[nH]c2)=O)C2CCC1CC(C(=O)NCC(C)C#N)C2 C1(C#N)(C(N2CC(CC(C)NC(c3ccn(C)c3)=O)C2)=O)CCCC1 c1(CCC)cc(C(=O)NC2CC(CCNC(=O)C=C(Cl)Cl)C2)cc(O)n1 c1(NC(C2N(C(CCN(C)CC)=O)CCSC2)=O)cc(OC)c(OC)cc1C C=CCCC(C(=O)C1CC2C(OCC)C(C(=O)O)C1C2)NC(c1cc(O)nc(C)n1)=O C1(O)(CCNC(CN(CC(=O)NC(C)C)C)=O)CCN(C(=O)C=C2CC2)CC1 N1(C(c2cccc(C(=O)NC3CC3)c2)=O)CC2CC1(c1cn(CCO)nn1)CO2 c1(C(=O)NCC2(F)CC(NC(c3cc(C)ns3)=O)C2)cn(C)nc1C(F)F c1(C(=O)NCCN(C(=O)CC2(C(F)F)CC2)CC)cc(S(N)(=O)=O)ccc1F N1(C(c2cn(C(C)C)nc2)=O)CC(C2CCN(C(C3CCCC(F)C3)=O)CC2)C1 CC(C)(C)CCCCC(=O)N1C(C(=O)NCc2nc(=O)o[nH]2)CC2CCCC12 N1(C(C(c2ccc(F)cc2)(C)F)=O)CCOC(CNC(c2cnc[nH]2)=O)C1 N1(C(CNC(C2C(C)C2)=O)=O)CCC2(C1)CN(C(c1c[nH]ccc1=N)=O)C2 C(c1ccc(Br)s1)=CC(N1CC(CNC(Cc2c(C)cco2)=O)C1)=O C1(NC(C2(C)CC3CCC2C3)=O)CN(C(c2ccncc2Cl)=O)C2(CCCC2)C1 C1(C(N(C(C)CNC(=O)CN(C2CCCCC2)C)C)=O)CCCS(=O)(=O)C1 c1(CNC(C2C(NC(c3c(COC)cc[nH]3)=O)CCCC2)=O)cc(C)cc(F)c1 CN1C(=O)Cc2ccc(C(=O)NCC(C)(C)CNC(C34CCC3CC4)=O)cc21 N1(C(C(CCCOC)C)=O)CC(NC(c2cc3sc(C)nc3[nH]2)=O)C2(CCC2)C1 C1(NC(C2(C)CC2Br)=O)CCC2CN(C(c3c[nH]c(C(F)(F)F)c3)=O)CC2C1 CC1CN(C(=O)CC(=O)OC(C)(C)C)C(C)CN1C(=O)CC1CC(OC(F)F)C1 Cc1ncc(C=CC(=O)NC2CC(N(C)C(C3CCCCS3(=O)=O)=O)C2)c(O)n1 C(=O)(CC1=NN(C)C(=O)C1)NC(COCC)C(=O)NCC(C)(C)OC(C)C N1(C(C)C)CCCCC1C(=O)NCCCCNC(=O)C(c1cccc(Cl)c1)O CCCCC(F)C(=O)NCC(C)(CO)NC(c1cncc(C2CC2)c1)=O N1(C(c2c(CC)nc(C(F)(F)F)o2)=O)CCN(C(=O)C(C)(C)CCl)CC(O)C1 S(=O)(=O)(c1ccn(C)n1)N1C2CN(Cc3cccc(C=C)c3)CC1C2 c1(C(=O)OC)ccc(C=CC(N2CCC(F)C(NC(C)=O)C2)=O)cc1F C1(C(=O)NC(C2(CNC(C3CC(OC)C3)=O)CC2)C)Oc2ccccc2OC1C c1(SCC(N2CC3C(NC(c4c(CC)occ4)=O)(C3)C2)=O)nnc2ccccn12 c1(NC(CC(CC)C)C)ccc(S(=O)(=O)NCc2ccncc2C(C)C)cc1F c1(CNc2cc(C)no2)c(F)ccc(Br)c1C.N12CC(C)CC1C2=O CCCCCC(C)(CC)C(=O)N1CCCCC(CNC(=O)CCCC(=O)NC)C1 c1(C(N(CC(C)NC(C2CC(CC(C)(C)C)C2)=O)C)=O)ccn(C2CC2)n1 N1(C(c2c(C)onc2)=O)CCCC2(CCC(NC(c3cn(C)c(O)n3)=O)C2)C1 C1(CC(=O)NCC2CCN2C(=O)C(O)C2CC2)CCn2cncc2C1 N1(CC)CC(NC(c2ccc(-n3cc(C(C)O)nn3)cc2)=O)C(C)C1 C1(NC(C(C(C)C)CCN(C)C)=O)CC2(CCCN(C(C3(C)CSC3)=O)C2)C1 c1(C(=O)NCCC(CNC(C=CCOC)=O)O)c(F)cc(F)cc1F C(=O)(CCCCCS(N)(=O)=O)NCCC1N(C(C(C)S(C)(=O)=O)=O)CCOC1 Cc1cnc(CC(=O)N(C2CCN(C(=O)CCOC(C)C)C2)C)[nH]1 N1(C(Cc2c(C)ncs2)=O)CC(NC(c2c(C)ccn2C)=O)CC12CCC2 C(=O)(C(F)CCCCC)NC(CCC#C)C(=O)N1CCC(CC2CC2)C1 c1(C(=O)NC(CCCNC(CC=CC)=O)C)cc2ccsc2n1C C1(CSC)CCCN1C(=O)CCCNC(=O)C(c1ccccc1)F c1(N2CCN(C)CC2CNC(c2ccc[n+]([O-])c2)=O)ncnc2c1CCO2 N1(C(C#CC2(C)CC2)=O)C2CCC1CC(NC(c1cc(C(F)(F)F)no1)=O)C2 c1(C(=O)NCC(C(C)(C)C)NC(c2c(C)con2)=O)cc(Cl)c2n[nH]cc2c1 c1(OCC)ccc(F)c(F)c1.C12N(CC1(C)C)C(=O)CN(C)CCCOC2.O.C C(CN(C(=O)CNS(=O)(=O)NC)C)(CO)(CO)NC(CN(CCOC)C)=O.C=O N1(C(c2cnn(C)n2)=O)CCC2(CCOCC2)C(NC(=O)CC(=O)NC2CC2)C1 c1(C(=O)NC23CC(C2)N(C(c2n[nH]cc2Cl)=O)C3)cnc(OCC(F)F)c(Cl)c1 C1(NC(C(C)(C)C)=O)CN(C(c2cc3ccoc3s2)=O)CC12CC2 N1(C(C2(OC(C)=O)CC2)=O)CCOC2CN(C(C34CC5CC(CC3C5)C4)=O)CC12 CC1CN(C(c2ccc(CNC(c3cccs3)=O)s2)=O)CC(C)(C)C1 C1(NC(CCCN(C(C)C)C(c2ccnn2C(F)F)=O)=O)CCCC1C#N CCC(CC)(CC)C(=O)N1CC(C(N2CCC(C)(COC)C2)=O)CCC1(C)C C1(CC=C)(NC(=O)C(O)CC(C)C)CCCN(C(=O)C=Cc2ccc(CC)o2)C1 N1(C(c2c(SC)cccc2)=O)CC(NC(c2nn(C)cc2SC)=O)CCC1C C(=O)(CC1=NN(C)C(=O)C1)NCC(CC(=O)NCC1(O)CCN(C)CC1)OC C1(NC(Cc2scc(C)n2)=O)CN(C(=O)CC2(C#N)CC2)CC2(CC2)C1 Cc1cn2cc(C(=O)N(C(C)CNC(c3cc[nH]c3)=O)C)sc2n1 CN1CCCCC1CC(N1CCC(C(C)(O)CNC(c2nccn2C)=O)CC1)=O C(C(C(C)(C)C)NC(=O)C(C)SC(F)(F)F)NC(C(CC)NC(N)=O)=O CC1COCC(CNC(N2CCC(Cc3nnn(C)n3)CC2)=O)O1 Cc1ccc(C(F)(F)F)cc1C(=O)NC1CC(C)N(C(=O)CCSCC(N)=O)C1 c1(NS(=O)(=O)CCCCl)cccc2c1CN(CC(F)(F)F)C2 C(CCC(O)C(=O)NC1CC(CO)N(C)C1)NC(c1c(CC)n(C)cc1)=O C1(NC(c2cc(C)c(C)o2)=O)CCC2CN(C(C3CCC4(CCC4)OC3)=O)CC12 c1(CC(COC)OCOC)nc(-c2ccc(F)cc2)nn1C12CCC(CC1)C2 N1(C(C(n2cc(CO)nn2)C)=O)CCN(C(=O)C(O)Cn2cncn2)C(C)C1 N1(C(CC(=O)NCC)=O)CCCC(C)C1CNC(=O)COCc1cc(C)on1 C1(NC(CCN2CCC(CN(C)Cc3ccccc3)CC2)=O)CCCCC1(C)C N1(C(C(C)OCC)=O)CCCC(C)C1CNC(=O)Cc1n[nH]c(=N)s1 c1(C(N2CC(C(C)NC(C(C=CC)O)=O)C2)=O)ccc2c(=N)[nH]cnc2c1 CN1CC=C(CCNC(c2cn(CCNC(C3CCCC34CC4)=O)cn2)=O)CC1 N1(C(CCCc2ccc(C)s2)=O)CCSCC1CCNC(C1C2CC3C(C2)C13)=O O=C(C(F)C(F)(F)F)N1CCC1C1CCCC1O.c12ccc(cc1)Cn1cc-2nn1 C(C(C(=O)NCC1(CO)CC(C)(C)C1)C(C)C)NC(CSCCC(C)C)=O c1(N(C)C)ccc(C(=O)N(C2CCN(C(c3sccc3F)=O)C2)C)nc1 c1(C(N2CCN(C(C34COCC3C4(F)F)=O)CC2)=O)cncc2[nH]ccc12 c1(C(N2CCN(C(CNC(C(C)CO)=O)C(F)(F)F)CC2)=O)nccc(N)c1Cl N1(C(C(CC)n2ccc(C3CC3)n2)=O)CCc2[nH]nc(I)c2C1 C1(=O)C(CC(C)C)N1.C(C(C)(C)N(C(=O)COCCN(C)C)C)SC c1(C(C)=O)cn(CC(=O)NCCCCNC(c2coc(C(F)F)c2)=O)cn1 N1(C(CCCN=[N+]=[N-])=O)CCn2c(CNC(C3CCCS(=O)(=O)C3)=O)nnc2C1 CC(O)CCCc1cn(C2(c3cccs3)CC2)nn1.C1(=O)CN1 CC1CCN(C(C2CC3(CCC3)CO2)=O)CCN1C(=O)Cn1cnnc1O Cc1cc(O)ncc1C(=O)N(C(C)C(=O)NCC1(C)CCCC1O)C C(C(CC(F)(F)F)NC(=O)CC=C(Cl)Cl)NC(c1occ(C)c1C)=O c1(CNC(C(C)NC(=O)Nc2cc(F)ccc2F)=O)cn2ccncc2n1 C1(C(=O)NCc2c[nH]ccc2=O)CC(F)(F)CN1C(c1ccc(F)c(F)c1)=O c1(-n2nc(C(=O)O)c(O)ccccc2)nc2ccc(F)cc2n1C(F)F C1(CNC(=O)CSc2cccs2)CSCCN1c1cc(-n2cncn2)ncn1.C(=O)C c1(NC(C(=O)NCC(CNC(CCC=CC(C)C)=O)(C)C)=O)ccc(C)c(C)c1 C1(CNC(Cc2c(C)non2)=O)CCN(C(=O)CCOCCN(C)C)CC1(F)F CCC1=C(C(=O)NCCC2CC(OC)CN2C(=O)CCCCN(C)C)SCCO1 c1(OC(CC)C)ccc(CNCc2ccc(CC)nc2)cc1 C1(O)(SC)CCN(C(=O)C(N2CCC(NCS(C)(=O)=O)CC2)=O)CC1.C(CC(C)C)O N1(CC)CCCN(C(=O)C(C2CCC2)NC(C2CC2C(C)(C)C)=O)CC1 CCC(CCC(=O)N1CC(=O)NC(C(C)C)C1)NC(=O)C(C)Cn1ccnc1 C=Cc1ccc(C(N2CC3CCC3(CNC(C3C(C)C3C)=O)C2)=O)cc1 N1(C(C2OCCN(C(C=CCOCCOC)=O)C2)=O)CC2(C1)CC(C)(O)C2 c1(C(N(CC(CNC(COCC(=O)OC)=O)(C)C)C)=O)ccc2c(c1)CCC=C2 C(=O)(CS(=O)(=O)C1CC1)NC12CC(NC(c3c(C)nc(C(C)C)cc3)=O)(C1)C2 CCC(C)C(C(=O)N(CC(c1nn[nH]n1)C)C)NC(=O)C(CN(C)C)CC C(=O)(C1=C(C)S(=O)(=O)CC1)N1CCCC(CN(C(C(F)OC)=O)C)C1 N1(C(C(C)CC2CCC2)=O)CCOCC(NC(=O)Cn2cccnc2=O)C1 c1(C(=O)NCC2CCN(C(c3c(C)cc(C(F)(F)F)s3)=O)C2)cccn(C)c1=O C1(NC(C2CCN(C(=O)OC)CC2)=O)CC2CCC(C1)N2C(=O)C1CC1 c1(C2C(C(N(CC(=O)OC)C)=O)C2)ccncc1.C1C(=O)N1C C1(CN(C)C(C2CCCN2)=O)CCCC1C(=O)NCCNC(N)=O c1(CC)cc(CC(=O)N(C)CCN(C(=O)C(C)NC(C2CCC2)=O)C)no1 N(C1CCCn2nccc21)C(C(CC(C)C)ONC(c1nc[nH]n1)=O)=O C#CCC(O)C(=O)N(C)CC1(O)CN(C(c2ccc(C(=O)N(C)C)cc2)=O)C1 n1(CC(N2CCC(O)(C(C)NC(=O)C(N)=O)C2)=O)c(=O)c(=O)[nH]c2ccccc12 N1(C(CC2CC(OCC)C2)=O)CCN(C(=O)CCN2CCOCC2=O)CC1CC C1(C(F)(F)F)(C(=O)NC(CNC(c2ccc(OC)o2)=O)C)CC2C=CC1CC2 C1(C)(OC)CCCN(C(C2CCCN(C(C3(F)CCCCC3)=O)C2)=O)C1 C=CC1(CC(N2CCSCC2CO)=O)CN(C(c2ccc(OC)o2)=O)C1 c1(C(N(CC(CNC(C2C(C#C)C2)=O)O)C)=O)c(C)cnc(OC)c1Cl CCC(CC(=O)NC1CC2(CC2)C1)NC(c1sc(C)cc1C)=O c1(CN2C(CCC(=O)Nc3cncnc3Br)CCC2)ccc(O)c2ncccc12 Cc1ccc2c(c1)CC(C(=O)N(C(C)CNC(=O)CCc1cccc(F)c1)C)S2 C=C(C)CCC(=O)NCCCC(C)NC(c1ccnc(N2CCOC(C)C2)c1)=O C(=O)(C1=CCSC1)NC(C1CCCCC1)C(=O)NCC1CC(C)C1 CCCCCCC(C)(C)C(=O)N(C)CC1CC(F)CN1C(C1CC1(C)C)=O C1(C(CO)NC(c2n[nH]cc2C2CCC2)=O)CCN(C(=O)C(O)CO)CC1 CCCCCC(=O)NC1CC(CCNC(=O)C(C)NC(C2CCCC2)=O)C1 C=C1CCC(C(N2CCC2C(=O)NC2CCN(C3CCOCC3)C2=O)=O)CC1 c1(N(c2nc(CCC(N3CCCC(CC4CC4)C3)=O)cs2)C)ccc(F)cc1 CC1(C)CCCC(CC(=O)NCC2(O)CCN(C(=O)CSc3nccs3)C2)C1 n1(C(CC(=O)OCCN(CCC)C(=O)NC)CC)cnc2ccccc12.COC C(=O)(C1=CNC2=NCCC2=C1)NC1CC(CNC(=O)CN2CCCCC2=O)C1 C1(CCNC(c2c(OC)nn(C)c2)=O)CN(C(=O)C=C2CCN(C)C2)CCCO1 c1(OC)cc(OC)c(CN2CCCC2(C)P(C)(C)=O)cc1-c1cn(C)nn1 C(=O)(C1=CCC(NC=O)C1)NCCCCN(CC)CC.c1(C2CC2)ccno1 C=CC(C)(CC)C(=O)NC(CNC(c1cc(OC(C)C)cc(Br)c1)=O)CO N#Cc1ccc(N)c(C(=O)NCCS(=O)C(F)(F)F)c1 C(C)(C(=O)NOC(c1ccccc1)C)N(C(c1ccc(C(C)=O)o1)=O)C Cc1oc(CO)cc1C(N1CCC(N(C(=O)CC2(O)CCOC2)CC2CC2)C1)=O c1(C(N2CC(C)C(NC(C3CC(=O)N(C)C3)=O)C2)=O)ccc2c(c1)CCC=C2 N1(C(=O)Cc2csc(Cl)n2)CC2OCCN(C(c3ccc4c(c3)NCC4)=O)C2C1 C(=O)(CCC(=O)N1CCCC1(C)C(=O)NCc1nc(C)c(C)s1)N(CCC)CCC C1(CN(C(=O)C(c2ccc(Cl)cc2)(F)F)C)COCCN1C(c1cnco1)=O O(NC(=O)CNC(=O)CC1CCOC1C)CC(=O)NCC1CC(OCC)C1 C1(C(=O)NC(CC(C)C)(C)CNC(c2cnnc(O)c2)=O)CCS(=O)(=O)C(C)C1 C1(OCC)CCCC1N=c1[nH]c(=NC(C)c2ccc(Cl)cc2C)c2sccc2[nH]1 n1(CC)ncc2c(N3CCC(F)(C(=O)Nc4cc(Cl)c(F)cc4C)C3)ncnc12 CC(C1OCCc2ccccc21)NC(=O)CCSc1ccc(F)c(F)c1 N1(C(c2ccnn2C2CC2)=O)CC2CCN(C(c3cccnn3)=O)CC2C1 c1(CCC)noc(CCC(=O)N(C(CNC(=O)CN(C2CC2)CC)C2CC2)C)n1 N1(C(c2c[nH]c(=NCC)s2)=O)CC=C(CCNC(C2CC(=O)N(C)C2)=O)CC1 Cc1ccc(-n2cc(NC(C3CCC(=O)O3)=O)cn2)cc1Cl C(C(C)(C)CC(=O)NCC1(O)CN(C(=O)CCCOCCOC)C1)OCC c1(C(=O)NCC2CC(NC(c3nc(C(C)=O)sc3)=O)C2)ccc(C#N)cc1 N1(C(CCC#N)=O)CC2(CCC2)CC1CNC(c1ccc(C2SCCS2)cc1)=O C1(C(F)(F)F)(C(=O)NC2CC(CN=c3[nH]nc(C)o3)C2)CC2CCC1CC2 N1(C(CC(C=C)CC)=O)CC(C)CN(C(=O)CCCc2ccccc2)C(C)C1 N1(C(C(CC)(C)OC)=O)CCCC(C2CC2NC(=O)CO)C1 c1(C(=O)NC2C(C)N(C(C3CC3(C)C(F)(F)F)=O)CC2)cccc(F)c1Cl c1(OC)cc(CC(=O)NCC(O)CCNC(=O)Cc2cnccc2OC)ccn1 C(=O)(C1CCCn2cnnc21)NC1C2CC(CNC(=O)Cc3cncs3)(C2)OC1 Cn1cc(C(=O)NC2CCCC2CNC(c2cnsn2)=O)nn1 C1(NC(C(COC)O)=O)CCN(C(c2ccc(-c3nnc(C)o3)cc2)=O)C(C)C1 CC(C)C(C(=O)NNC(=O)NCC1CN(C)CCN1C)N(C)C c1(C(N2C(CN(C)C(c3cc(O)nc(O)n3)=O)CCC2)=O)cc(Cl)c(F)cc1F n1(C(CC)C)nc(-c2ccc(N3CCCC3)nc2)nc1C(C)OC1(C)CCC1 C(C(C)(O)C(=O)NC1CCC1CNC(c1cnn(C(C)(C)C)c1N)=O)OC CC1(C)CC(C(=O)NCCN2CCC(NC(=O)CCOCC3CCC3)CC2)CO1 C1(NC(CC)=O)CCCCCC1NC(=O)CCCN1C(=O)CCC1=O c1(C(N2C(COC)CN(C(C3CCSC3)=O)CC2)=O)cc(F)cc2cccnc12 CCC(C)C(C(=O)NCC1(C(=O)Nc2cc(C)sc2C)CC2(CC2)C1)OC C1(OC)CCN(C(c2ccc(CNC(c3[nH]cc(C)c3C)=O)nc2)=O)C1C1CC1 Cn1ncc2c1CC(NC1COC(C)(C)C1)CC2 C(CCCCC(=O)NCc1nnc(O)o1)N(C)C(C1(CN(C)C)CCC1)=O c1(CC)cc(CC(=O)NC(C)CNC(=O)CC(c2c(C)noc2C)C)n(C)n1 c1(C(N2C(CNC(C3CC(OCC)C3)=O)COCC2)=O)ccc2c(c1)OCCN2 c1(C(N2CCCCC(N(C(C3CCN(C)C3)=O)C)C2)=O)cccc2nc(Cl)cn12 Cn1cnn(CC(=O)NC2(C(=O)NCC(C)(C)C3CCC3)CCCC2)c1=O C(CCC(=O)NCC1C=CCN1C(c1c[nH]c(=N)o1)=O)N(C)C c1(C(C)C)cc(NCCN2CCCCC2)ncn1.c12noc(n1)CCCNC2=O CC1C(CO)CCCN1C(=O)CCCCN(C)C.c12ccc(c(F)c1)CNC2=O N1(C(CCC(=O)N(C)C)=O)CCCCC(C2CN(C(=O)CC3CCCCO3)C2)C1 CC1CCN(C(C2CC(C(F)F)C2)=O)CCN1C(=O)Cc1ccsn1 C1(c2ccc(NCC(c3ccccc3)C)cc2)(C(=O)OC)CCOCC1.C(C)C N1(C(c2ccc(C)c(C)n2)=O)CCOC2CCN(C(C3CCC(C)(C)C3)=O)CC12 C(=O)(C(CO)C(F)(F)F)N1CCC(n2cc(-c3cccc(N)c3)nn2)C1 C1(CC(=O)N(C(C(=O)OCC)COC(C)C)C)CC(N)CC(C)(C)O1 N1(C(C)=O)CCNCC1C(=O)NCC1(Nc2cccc(Br)c2)CCCC1 Oc1nc2ccc(-c3nc(C4CCCCC4)nn3-c3ccccc3)cc2[nH]1 C1(CNC(C2C(c3n(C)ccn3)C2)=O)CC(NC(c2cccc[n+]2[O-])=O)C1(C)C O=C(CCC(F)F)Nc1cnc(OC2CCN(C(=O)COCCF)C2)cn1 N1(CC(=O)Nc2nc(-c3ccccn3)n[nH]2)CCC(NCCC(O)C2CC2)C1 C#Cc1cnn(C)c1C(=O)NC1CCC(C)N(C(=O)Cc2cccnc2)C1 CCCCC(O)C(=O)N1CCC(C2N(C(=O)C(C)C(C)C)CC2(C)C)CC1 Cc1cc(CCCC(=O)NC2CCC2NC(=O)C(C)C2(O)CCC2)c(C)s1 CCCCCCCCCCCC(O)C(=O)N(CCC(C)NC(=O)C=CBr)C c1(C(=O)NC2C(CNC(C3(C)COC3)=O)C2)ccc(F)c(F)c1F c1(C(=O)NCC(C)(CO)NC(Cn2nc(C)oc2=O)=O)cc2c(Cl)cncc2s1 CC1CC(CNC(c2ccc(Cl)nc2N)=O)CCN1C(=O)C=Cc1ccco1 CC1CC2CN(C(=O)CC3CCCNC(=O)C3)CC2N1C(c1ccc(Cl)o1)=O C1(C(=O)NCc2cc(C)c(C(=O)NC3CCN(C(C)C)C3)o2)CCOC(C)(C)C1 C1(c2ccccc2)(C(=O)NC2CC(CNC(C=C(COC)C)=O)C2)CCCC1O CC1(C)CCN(C(c2ccc(CO)cn2)=O)CC1CNC(C1CCC12CCC2)=O C12(NC(C3=CNS(=O)(=O)N=C3C)=O)CC(C)(C1)OC21CN(C(=O)CSC(C)C)C1 N1(C(CC(CCC)O)=O)CCC2(CCN(C(=O)CC(C)(F)F)C2)C1 C1(CC#C)(C(N2CCOC(c3cn(CC45CC(CO4)C5)nn3)C2)=O)CCCOC1 c1(CC(=O)N(CC(C)NC(=O)C=C2CCCCC2)CC)ccc(Br)c(OC)c1 c1(C(=O)NC(CC)CNC(=O)C(CC2CC2)OC(C)=O)c(C)ncnc1C c1(CC)noc(C)c1CNC(c1sccc1CNC(C1COCC1(C)C)=O)=O C1(COC(C)C)CN(C(=O)CN2CCOCC2=O)CCO1 C=C1CCC(C(=O)N(CCC(C)NC(C)=O)C)CC1.C1(=O)CCCN1.C(C)(C)(C)S c1(CC(=O)NCC2N(C(C3C(=C)C3)=O)CC2)nncn1C(C)C c1(CN2C(Cc3nccc(O)n3)CCCC2)n[nH]c2c1CCCC2 N1(C(CNC(c2n(CC)ncc2)=O)=O)CCCN(C(=O)CNC=O)CC1C O=C(C1CCCn2cnnc21)NC1(CNC(C23CCCCC2C3(F)F)=O)CC1 N1(C(C(CC=C)CNC(c2cc(C)ccc2F)=O)=O)CCCC2(C)CCCC12 C1(OC)CCC(C(F)(F)F)N(C)C1.c12ccc(cc1)C(=O)Nc1ccnn1-2 N1(C(c2cc(C(=O)OCC)c(C)[nH]2)=O)CCN(C(c2ncc(Cl)s2)=O)CC(O)C1 c1(OC)nc(Cl)c(C(=O)NCC2CC(NC(=O)C(C)Cc3ccccc3C)C2)s1 c1(N(C)C)ccc2c(c1)CCC(CNC(=O)NCc1csnc1OC1CC1)O2 C1(NC(=O)CC(F)(F)Cl)CN(C(=O)CCOC2CC2)CC12CC2 c1(C(=O)NCC2(CNC(CCc3onc(C)n3)=O)CC2)ccnnc1O c1(CN2CCC(C)(C(N(CCCC)CCCC)=O)C2)cc(Cl)cnc1F N1(C(c2nccnc2C)C(=O)NCCOCC)CC(=O)N(C)CC1CC C1(CC(=O)NC2CC(CNC(C3C(C(C)=O)C3(C)C)=O)C2)CCCC(C)(C)C1 CN1CC(C)(C(N2CC(CNC(=O)CC3(CO)CCCC3)C2)=O)CCC1=O c1(C(=O)NC2(C)CCN(C(C(CC)(C)C#N)=O)C2)cccc2c(Cl)c(Cl)sc12 C=CCCCCCCCCC(=O)NCC1CCCN1C(C1(C)CC1(F)F)=O CCC(O)CCN=c1[nH]c(=NCc2cnc(C)o2)[nH]c2cccnc12 C1(NC(c2sc(CC)c(C)c2)=O)CC2(CCN(C(C3CCC(=O)N3C)=O)C2)C1 Cc1cc(Br)ccc1NC(N1CCN(C(=O)OC(C)(C)C)CC1)=O.C1CCO1 c1(CN2CC(CC)N(c3nc(C)ncc3C#N)CC2)cccc2ncccc12 Cc1ccc(-n2nc(Cn3cccn3)nc2-c2[nH]nnc2C)cc1 Cc1cc(=NC(C)CN2CCCCCC2)[nH]c(=NCCC(F)(F)Cl)[nH]1 C(=O)(C(CSNc1ccc(CSC)cc1)OC(C)=O)OC c1(NC(C)=O)ccc(C(=O)C(N2CCC(N(C(=O)C(C)O)CCO)CC2)=O)cc1 N1(C(CCCNC(=O)NC)=O)CC2(CC=CC(C(=O)OC(C)(C)C)(C(=O)OC)C2)C1 c1(C(N2CCC(N(C)C)CC2)=O)cc(-c2cccc(Br)c2)cnc1O N1(C(C2CCC(N(C)C)CC2)=O)CCN(C(=O)CCC(F)F)CC(C)(C)C1 c1(C(=O)NC(CC)CNC(=O)CCSC)cnc(C(C)(C)C)nc1C C1(C)(C(=O)NCCCCNC(C(=Cc2cccs2)C)=O)CCOCC1 n1(CC)cc(Cl)c(C(=O)NCC2C3CN(C(=O)C=CC(C)(C)SC)CC23)n1 c1(C(C(N2CC(NC(C(C)(C3(C)CC3)OC)=O)C2)=O)C)cccc(O)c1 C1(C(N2CC3CN(C(C=C(CCC)C)=O)C3CC2)=O)Cc2c(C)cccc2O1 c1(C(=O)NC(C2CCCN2C(c2nnsc2N)=O)C)ccc(C2CCOC2)cc1 N1(C(C2CC(CC)C2)=O)CCn2ncc(CN(C(=O)CSc3cccs3)C)c2C1 c1(C(=O)NC2CN(C(C(C)(F)F)=O)CC2O)ccc(Br)c2c1OCCC2 C(CC(CC)C(=O)N(CCC(=O)NC1CCCC(N(C)C)C1)C)=CC c1(CC(=O)NCC(C)CN(C)C(C2C=CCCC2)=O)cccc(F)c1O c1(C(=O)NC(C)CCCNC(=O)C(C)(C)OCC(F)(F)F)cnn(C)c1N C1(CNC(=O)Cc2ccncc2Cl)CCN(C(=O)C=CBr)CCO1 C1(CNCC2(O)CCC(Cc3n(C)cnn3)CC2)CCn2ccnc2C1 C1(NC(=O)NC)CC(C(=O)N(CCCNCC(=O)OC(C)(C)C)C(C)C)C1 c1(C(N2CCC(NC(C(CCCC)CC)=O)C2)=O)ccc(=NCCOCC)[nH]c1 C1(NC(=O)CCCCN2CCCC2)CN(C(C23CCC2C3)=O)CCC12CCC2 CC1C(c2ccc(F)c(Br)c2)OCCN1CC(C1CC(C)(C)C1)=O N1(c2nccc(SC)n2)CCCC2C1CCN2C(c1ccn(C(F)F)n1)=O N(C1CC2(CCC2)Oc2ccc(F)cc21)S(=O)(=O)CCc1ccccn1 C12(C(N3CCC(CNC(C=CCC)=O)C34CC4)=O)CC3CC(C1)CC(F)(C3)C2 CC(CCC(=O)NCC12CC(NC(c3ccc(O)cc3)=O)(C1)C2)S(C)(=O)=O N1(C(c2ccn(CC)n2)=O)CCC(NC(c2cnc(SC)nc2O)=O)C(F)C1 c1(NC(C(=O)OC)(C)C2CC2)ccc2oc(Cl)cc2c1 CC1(C)CCN(C(c2ncccc2O)=O)C1C(=O)NCC1CC(F)(F)C1 c1(N)ccc(CN2CCCCC2)cc1.C1(NC(=O)C(=O)NC)CC2CC2C1 C1(CNC(c2cc(C)oc2)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1(F)F c1(CC(=O)N(CCCNC(=O)C(C)(C)C)CC)c(OC(F)F)cccc1Cl.C(C)(=O)N CC1(C)C2CN(C(C34CC3CCN4C(=O)CC3CCCSC3)=O)CC12 C(=O)(C(F)C(C)C(F)(F)F)NCC(C)N(C(c1ccc(CC)cc1OC)=O)C c1(C(=O)COC(=O)CCCC2CC2)cc(F)c(Br)c(F)c1 S(=O)(=O)(c1nnn(C)n1)NC(c1ccc(F)cc1)c1ccc(C)o1 C1(NC(c2nccc(N)c2Cl)=O)CN(C(=O)COC2CCOC2)C2(CCC2)C1 C1(C(=O)NCC(C(=O)NCC2OCCN(CC)C2)C)CC(=O)NC(=O)C1 c1(N2C(CNC(CC(C)C(F)(F)F)=O)CC(F)(F)C2)ccc2c(n1)CCCC2=O C1(CNC(c2c(C(C)C)occ2)=O)CN(C(C2(C(F)F)CCC2)=O)CC12CC2 C1(COC)CN(C(=O)C(Cl)=CCl)CCN1C(=O)C1=CSCS1 c1(CC)ncc(C(=O)NCC#CCNC(=O)Cc2nc(C)sc2Cl)c(C)n1 C1(NC(C2(CNC(C3C(C)(C)COC3)=O)CC(CO)C2)=O)CC(C2CCC2)C1 c1(CN(C)C)ccncc1C(F)(F)F.C12(OC)CN(C1)c1nnc(o1)C2 c1(C(N2CCC(C)C(NC(c3csc(CO)n3)=O)C2)=O)cc2n(n1)CCCCO2 C(=O)(C1OCCc2cc(O)ccc21)NC1(CNC(C(C)C(C)(F)F)=O)CC1 C=C1CC(C(=O)N(C)C(C)C)(CNC(C2(SC)CC2)=O)C1.C1CCN1.COC C(CC(C(=O)NCC1CC(C)(O)C1)NC(=O)CC1CCN(C)C1=O)OC c1(OCC)cc(-c2cn(C3CC(C(=O)Nc4cnc[nH]4)C3)nn2)ccn1 c1(NC(C)=O)cccc(C(=O)NC(C)CC(C)NC(=O)C(C(C)O)N(C)C)n1 Cn1cnc2c1CCCC2C(=O)NC1CC(NC(=O)CCn2cccn2)C1 CC(C)C(C(C)NC(=O)Cn1cnnn1)NC(c1cc(C#N)no1)=O C1(C(N2CCCC(NC(c3ccn(C4CC4)c3C)=O)C2)=O)(OC)CCS(=O)(=O)C1 c1(N2CCC(COC)CC2)nc(NCC(C2CCCCC2)C)c2ncn(C)c2n1 CCC(C(=O)NCC1(O)CN(Cc2ccc(Cl)c(C(=O)NC)c2)C1)C(F)(F)F N1(C(C2C(C)(C(C)C)C2)=O)CCC(NC(c2c[nH]ccc2=N)=O)C2(CCC2)C1 N1(CC2(CC(N3CC(O)(CNC(C4(CO)CC4)=O)C3)=O)CC2)CCOCC1 N1(C(c2c(C)[nH]cc2)=O)CC2OCCN(C(=O)CC3CCOC3)C2C1 CC(C)(C#N)CCC(=O)N1CCC2(CC1)CC2CNC(=O)Cc1ccsc1 C12(C(N3C(C)C(O)CC3)=O)CCCC1CCN2C(=O)C(Cl)Cl N1(C(C(N2CCCC(OCC)C2)=O)=O)CCCN(Cc2ccccc2)C(=O)C1 O=C(CCCc1cn(CCSC2CC2)nn1)NCS(=O)(=O)Cc1csc(Br)n1 CCCCCCC(C(=O)NC(CNC(=O)C=Cc1ncc(C)[nH]1)CC)NC(C)=O C1(C2CCCC2)(NC(C2C(C)(C)C(NC(=O)C(F)F)C2)=O)CC1 CCC(C)CCCC(=O)N1CCC2CC2(C(=O)N(c2cccc(C)c2)C)CC1 C(CC(=O)NC1CC2CC1CC2CO)(C(F)(F)F)NC(c1cc(C)nnc1O)=O c1(C(=O)NCc2cccc(OCC)c2)cc(F)cc(N)c1N c1(C(C(=O)NCC2CCN2C(c2nocc2Br)=O)OC)ccc(F)cc1 c1(CC)ncnc(N2CCC(NC(=O)C(c3ccc(Br)cc3)OC)C2)c1F C(=O)(C(CC(C)C)N(C)C(c1nonc1C)=O)N(CC(CC)CC)CC C#Cc1cnc(C(N2CC3CC(NC(c4sccc4Br)=O)C2C3)=O)c(C)c1 CCC(C(=O)OC)C(=O)NCc1n[nH]cc1C(=O)NC1(CC)CC1 N1(C(C2(CC#C)CCCO2)=O)CCN(C(=O)CCCOCC)C(c2cn[nH]c2)C1 C(=O)(CCCCCCNC(=O)C(C(C)C)SC)NCC(CC#C)(C)CO C1(NC(CC(C)N(C)C)=O)CC(F)CN(C(=O)Nc2cccc(Br)c2Cl)C1 c1(C(=O)NC(CC=C)CNC(=O)CCC2CCC(=O)NC2)csc([N+](=O)[O-])c1 N1(C(CNC(CC)=O)=O)CC(CNC(=O)CSc2ccc(Br)o2)C(C)C1 C(=O)(C(O)CCCNC(=O)CCc1nncs1)N1CCCC(OC)C1 C(=O)(CC(O)CC(C)(C)C)NCC(C)N(C(c1cc(C)cs1)=O)CC c1(C(C)C(=O)NC2CCC2CNC(=O)COCc2nc[nH]n2)c(F)cccc1F N1(C(c2nnn(C)n2)=O)CCC2(NC(=O)CCN3CCCCC3)CCCCC12 n1(CC(N2CC3C(CNC(C(C)O)=O)(CC3)C2)=O)ccc2ccc(F)cc12 Cc1cc2cc(C(=O)NOc3cccc(C(O)C(F)(F)F)c3)[nH]c2cc1F C1(NC(c2c(C)nsc2)=O)CCN(C(C2(C)CC=CC2)=O)CC1CO c1(CS(=O)(=O)NCc2n(C)nnc2)ccc(F)nc1 Cc1cnc(Cl)c(S(=O)(=O)NCCNC(C2CCC(c3ccccc3)C2)=O)c1 C1(C(C)(C)C)CN2CCC1(NC(=O)NC1(c3ccccc3)CC1(F)F)C2 C12CC3(CCC3)CN1C2=O.N1(C(CN(C(CSCC)=O)CC)=O)CCCC1 C1(NC(C)C)CCN(C(=O)Cn2ccnn2)C(C)C1.C12(CC1)C(=O)N2 O=C(CS(=O)(=O)N1CCOCC1)NC(Cc1ccco1)C(=O)Nc1ccccc1 C1(N(C(C2CN(C(C)C(=O)N(C)C)C2)=O)CC)CCOC(C)(C)C1 c1(C(=O)NC(CC=C)CNC(C2(C)CC2C(=O)OC)=O)cc(C)c(Cl)cc1F CCC(CC)C(C(=O)N1CC(C)(OCC(N2CCC3CN(C)CC23)=O)C1)OC Cc1ccc(C)n1CC(=O)NC(CCc1nn[nH]n1)C(=O)NCc1cnccc1Br C1(C(C(=O)N)NC(=O)OC(C)(C)C)CC(N(C)CC)C1.C1(=O)CCO1.C(C)(C)(C)O c1(C(=O)NCC(C)CN(C)C(c2nc[nH]c2C(C)(C)C)=O)ocnc1C1CC1 c1(N(C(c2ccccc2)CO)Cc2ccccc2)ccc(Br)cn1 C1(Cc2scc(COC)n2)CCCCN(C(=O)CCCNC(=O)C(C)(C)C)C1 C1(NC(C(CSC)OC)=O)CCN(C(c2cccc(N)c2F)=O)C1(C)C C1(C(N2CC(C(C(=O)NC(CCOC(C)C)C)O)C2)=O)CCSCC1 c1(CN2CC3(N(C(C(CCC)C)=O)CC3)C2)cc(OC)nc(OC)c1 CC1=C(C(=O)N2CCN(CC(C(=O)Cc3cccc(C)c3Br)=O)CC2)CCO1.O C(=O)(C1=C(Cl)CCOC1)N(CCCNC(C1C2(CC(OCC)C2)C1)=O)C C1(NC(=O)CSc2ncc[nH]2)CN(C(=O)CCSCC2CC2)CC1O c1(CC)cccc(C(=O)NC(CNC(c2ccco2)=O)C2CC2)n1 n1(CC(=O)N(C)CC2CN(C(C(=O)NCC)=O)CC23CC3)cnc2c1CCCC2 c1(C(=O)NC(C(=O)NC(C=C)(C)C)Cn2cccn2)ccc(F)c(O)c1 c1(CN(C(=O)C(C2CCCC2)NC(=O)CC2CCCC23CC3)C)cc(=O)cc[nH]1 C1(C(=O)NCC(CC)NC(c2cccc(Cl)c2O)=O)CCCC2CCCCC12 N1(CC(=O)NC(CNC(C2C(CCOC)C2)=O)(C)C)C(=O)NC(C)(C2CC2)C1=O Cc1ccc(C(CNC(=O)Cn2cnnc2)NC(C2CCC(F)(F)C2)=O)cc1 N1(C(c2c(OC)ccs2)=O)C2CCCC1CC(NC(c1cccn1C)=O)C2 C1(C(=O)NC2(CC=C)COC2)CCC(C)(C)CC1c1ccccc1 c1(C(=O)NCCOC2CCN(C(c3ccc(CC)[nH]3)=O)C2)cc(C)c(C)nc1O C1(C(=O)NC(C2CCN(C(Cn3c(C)cnc3)=O)C2)(C)C)CN2CCN1CC2C c1(CC(=O)NCC2(CC(=O)NC(CCOC)C)CC2)cncn1C CCCCC(CC)C(=O)NCC1CCCN1C(c1n[nH]cc1Cl)=O N1(C(C=CCC)=O)CCN(C(=O)C(CC)OC)CC1CCOCCOC C1(CC)C(=O)NCCN1C(=O)C(N1CCOC(c2cc(C)ccc2C)C1)=O N1(C(CC2(OCC)CCC2)=O)CCOCC1CCNC(=O)CN1CCCNC1=O c1(SC)nc(C(N2CC3(CC3)CC2CNC(C2CC2(C)C)=O)=O)c2ccccn12 C(=O)(CC(C)(C)CC)NCC(c1ccc(F)cc1F)NC(C=CCC)=O c12cc([nH]n1)C(=O)NCC#CCNC2=O.c1(CC2(SC3CC3)CC2)ccccc1 C1(NC(C(C)C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)C12CC2 Cc1[nH]nc(C(=O)N(C)CC2CCCN2C(=O)CCCc2n[nH]c(=N)s2)c1Cl c1(C(=O)NCC2(O)CN(C(C3(CC(F)F)CCCCC3)=O)C2)csc2nnsc12 C1(C(N2C(C(C)NC(c3ccncc3CO)=O)CCCC2)=O)CC(=O)NC(C)C1 CC(C)CC(C)(C)C(=O)N1CCC1Cn1cc(-c2cncc(F)c2)nn1 C1(NC(C2C(CC)C2)=O)C=CC(CNC(c2cncn2C)=O)C1 C1(C(=O)OC(C)(C)C)(C(=O)OCc2cnc(C(C)(C)C)o2)CCCCO1 N1(C(C=C)=O)CC2CC(C1)CN(C(N1CCCOC(C)C1)=O)C2 N1(C(C(C)(C)OCC(C)C)=O)CC2C(NC(c3ccc(O)cn3)=O)C2C1 C1(C(=O)NOCC=CCl)CC2(CCC2)CN1C(c1cc(O)cc(=O)o1)=O CC(C)(CC(=O)NCC1CCC(NC(C2(C)CC2C(F)(F)F)=O)CC1)C(F)F C1(C)(COC)CC(NC(=O)C=CSC)CN1C(=O)Cc1ccc(C(C)(C)C)cc1 C1(NC(C2CCC(C)(C)OC2)=O)CN(C(=O)CC2CC(F)(F)C2)CCC12CCC2 C(C(C(=O)NCc1occc1C(=O)Nc1cncn1C(C)C)NC(C)=O)OC C(CCC(C)(C)C(=O)NCC1(CO)CC1(C)C)NC(C1(OC(C)=O)CC1)=O CC(C)(CCCO)C(=O)N1CCC(N2CCN(C(=O)CCCNC(N)=O)CC2)CC1 c1(CC)nn(C)c(C(=O)NC2CCCN(C(=O)Cc3c(C)cccc3F)C2)c1Cl Cc1nc(C(C)(C)C)c(C(=O)NCCCCC(C)NC(=O)C(O)CN(C)C)s1 C(CCC(C(=O)N1CCOC(CN(C)C)C1)NC(C1CCOC1)=O)OC C(C)(C(=O)N1CCCCCO1)SCC(CC)C(C)C C1(O)(C(C)NC(c2cccnc2C2CC2)=O)CCN(C(c2ccccn2)=O)CC1 C(C(CC(=O)NOCC1CCOC1)C1CCC1)NC(C1(F)CCOC1)=O N1(C(C2(CCCC)CC2)=O)CCCC(CNC(c2conc2C2CCC2)=O)C1 N12CCC(C)(C1)CNC(=O)COCCC(Cl)=CC2=O.C(C(C)(C)C)N(C)C N1(C(C2CCCC23CC3)=O)CC2CCCC2(NC(C2(CO)CCC2)=O)C1 c1(C(=O)NC2CN(Cc3ccc(C)nc3)CC2F)ccc2nncn2c1 C1(NC(C=COCC)=O)(CNC(c2ccc(O)nc2)=O)CCCCC1C C1(N(CCOC)C(=O)OC(C)(C)C)CCN(N2CCCC2C2CCOCC2)CC1 C1(NC(C2OCCN(C)C2)=O)CCC(C)(CNC(c2cn(CCO)nn2)=O)CC1 c1(C(N2C(C)CC(NC(CN(C(C)=O)C)=O)C2)=O)ccc2c(c1)OC(C)(C)O2 N1(C(C(CC)C#N)=O)CCN(C(=O)Cc2ccc(Br)cc2C)C2CCCC12 N1(C(Cc2cc(C)ns2)=O)CC=CC(NC(=O)CC(=O)OC(C)(C)C)C1 CCCC(C(O)C(=O)NC1CC2(C1)CC(O)C2)NC(=O)CCc1ccccc1 c1(C(=O)NCC2CCN2C(=O)C(c2ccccc2)O)c([N+](=O)[O-])cnn1CCO CCC(C)(C)C(O)C(=O)N1CC(O)(CNC(=O)Cc2occc2C)C1 N1(C(c2c(OCC)oc(C)n2)=O)CCC2C(C1)CN2C(C1CCN1C)=O N1(CC(=O)N(C2CCN(C(=O)CCCCN(C)C)CC2)CC#C)CC2C=CC1C2 N1(C(c2coc(O)n2)=O)CC2CC(C1)N2C(C1CC2CCC2C1)=O CC(C)CC(C)(CNC(=O)C(C)(C)CF)NC(=O)Cc1cnns1 CCCC(CCC)C(=O)N1CCC(C)C1C(=O)N(C1CCOCC1)C C1(C2CN(C(C3CCNC(=O)C3)=O)C2)(NC(C(C)Cn2ccnc2)=O)CC1 c1(CNC2CCN(C(C3(C(N)=O)CC3)=O)C2)ccc(F)c(C(F)(F)F)c1 n1(C(C)C)cncc1C(=O)NCCN(C(=O)CC1(c2ccon2)CC1)C1CC1 CS(=O)S(=O)CCN=c1[nH]c(N2CCC(Cc3ccncc3)C2)nc2ccsc12 c1(SC)ccc(C)c(C(=O)NCCC(C)(C)NC(=O)Cn2cccc(O)c2=O)c1 CCCCCCC(CC)C(=O)NCC(C)NC(c1ccc(-n2cccc2)cc1)=O C1(CC(N2CC(O)(C(C)NC(=O)CCN3CCCC3=O)C2)=O)(CO)CCOCC1 N1(C(CC(CC)c2ccccc2)=O)CCC2(CCCN2C(=O)CC=C(C)C)C1 c12ccc3c(c1[nH]c(=O)c1cc(OC)ncc21)OCO3.c1(CC)c[nH]nc1C CC1CCOC1C(=O)NCCn1cc(CNC(c2ccc(Cl)s2)=O)nn1 c1(CCN=C(N(C)Cc2cnn(C)n2)NC2CC2)cc2c(cc1[N+](=O)[O-])OCO2 c1(C(=O)NCCN2CCOCC2)cc2c(s1)CCN(Cc1cccc(O)c1O)C2 Cc1cc(F)ccc1C(=O)NCC1CCN(C(=O)CCN(C)C)C(C)C1 c1(C(=O)NCC2C=CC(NC(C3C(OCC)C3)=O)C2)cc(CC)cc2c1OCC2 N1(c2ccc(CC(=O)OCC)cn2)CCC2(NC(C3CC3F)=O)CCCC12 c1(CCC)nc(C(=O)NC(C)(CNC(=O)CSc2cccs2)C2CC2)cs1 N1(C(C(CC(C)C)O)=O)CCC2(CCC2)C(CNC(=O)C#CC(C)(C)C)C1 C12(CNC(CC=C(C)C)=O)CC(NC(=O)Cn3c(C)nnc3S)(C1)C(C)(C)O2 c1(CNCCNC(C=CC(=O)OCC)=O)cc(C)c(NC(=O)C(F)C(C)C)o1 C(=O)(CCCC(=O)NC(C)C(C)(C)C(=O)NC1CCC1)OC CCC(CNC(=O)C(O)CNC(=O)C=Cc1cc[nH]n1)C(C)(F)F C(c1cccc(Cl)c1)=C(C)C(=O)NCCCCCNC(C1CC(C(C)(C)C)C1)=O C(=O)(C(O)C1=CCCCC1)NC1(CCC(N2CC(C)(CO)C2)=O)CCCC1 c1(CC(C)(C)NC(CCS(=O)(=O)NC)=O)ccc2c(c1)OCCO2 CCC(C)(C)CNC(C1(F)CN(C(=O)Cc2cscn2)C1)=O C1(C(=O)NC2C(CNC(C(C)SC(F)(F)F)=O)COC2)C2CCCCC12 C(=O)(C(C)CC(F)(F)F)NCC(CN(C(c1ccc(COC)o1)=O)C)(C)C C1(C(N(C2C(OC)COC2)C)=O)CCCCCN1C(c1ncnc(C)c1C)=O C(=O)(CC(F)(F)Br)N(CCCNC(=O)C=C1CCOCC1)CC c1(OC)nc(C(=O)NC(CNC(c2cn(C(C)C)cn2)=O)C2CC2)sc1C C1(CCC)CN(C(c2cn3ccnc3s2)=O)CCN1C(=O)C(=Cc1cnc[nH]1)C C1(=O)CC(C)(O)CN1.CCC(CNC(c1cnn(CCF)c1)=O)CO CC(C)P(=O)(CC(=O)NCC(c1ccccc1Br)=O)C(C)C c1(C(=O)OC)ccncc1OC1CCOC1.c1(C)ccnc(CO)c1 c1(NC(C2N(S(CCCC)(=O)=O)CC(O)C2)=O)cnc(C#N)c(C)c1 c1(NC(CC)C(C)C)ncccc1S(=O)(=O)NCCCCC1CC1 C#Cc1cc(C(N2CCC(CO)C(NC(=O)CCOCCOC)C2)=O)cc(F)c1 c1(C(=O)NCC2(NC(=O)CCc3ccccc3F)CCOC2)ccc(=O)oc1 C1(C(N(CCOCC#C)C)=O)CC2CN(C(=O)C#CC3CCCC3)CC2C1 Cc1ccc(CN2CC(NC(c3cccc(Br)c3)=O)CC(F)(F)C2)cc1[N+](=O)[O-] c1(C(C2C(c3nc(C(C)C)sc3)C2)=O)ccc2c(c1)OCCO2 Cc1cc(C(N2CCOC(C(=O)NCCN3CCCCC3)C2)=O)ccc1[N+](=O)[O-] CC1CCN(C(C2CCC3CC2CO3)=O)CCN1C(c1csnn1)=O Cn1nnc2ccc(C(=O)NC3CN(C(C4(CF)COC4)=O)CCC3(C)C)cc12 N1(CC(=O)N(CCNC(CC2C(OC)CC2)=O)C)C(=O)NC2(CCOCC2)C1=O C1(NC(CCSC)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)CCC1CO C(N=c1cc(F)nc[nH]1)C1CN(C(C23CCC(C2)OC3)=O)C1 N1(C(c2cnc(C)nc2)=O)CCC(C2CC2)C1C(=O)N(C1CCOC1)C CCCC(C)(CC)NC(C1(CC)CCN(C(=O)CC2CCCO2)C1)=O c1(-n2c(C)cc(C)n2)ccc(N(C(c2cc(O)n[nH]2)=O)CC2CCC2)cc1F C1(C(N(C2CCN(C(C3C(C)OCCC3)=O)C2)C)=O)C2CCC3(COC(=O)C13)O2 N1(C(=O)Nc2ccoc2)CCCC1C1CCCCN1C(=O)COCC(F)F C1(C(=O)OC)CC(C)N1C(=O)C(O)CNC(=O)CC1CC1 C1(NC(=O)C(c2cccc(Cl)c2)O)CC12CCN(C(C1CCCC(=O)O1)=O)CC2 c1(CN)ccc(C(=O)N(C)C)cc1.c1(C(CC)=O)nccs1 C12(NC(=O)CCc3ccc(F)cc3)CCCC1N(CCC(=O)NC1CC1)CC2 N1(C(C(CSC)OC)=O)CCC(C(=O)NCCC2CCOC2(C)C)C(O)C1 C(=O)(C1CCCc2nc[nH]c21)NCCCNC(c1cc(C#C)c(Cl)cc1)=O c1(C(=O)NC2C(OC)CN(C(C3CCCNS3(=O)=O)=O)C2)ccc(N)c(F)c1F N1(C(c2c(O)ccc(OC)c2)=O)CCC2(CC1)CC2CNC(=O)CCCOC O=C(N=c1nc2cccc(Cl)n2[nH]1)Nc1c(F)cccc1F.N12CCCC1C2 c1(NC(C(CNC(C(CC(C)C)OC)=O)(C)O)=O)c(C)nc2ncnn2c1C C(=O)(CCCCNC(C1CN(Cc2nc(Br)cn2C)CCS1)=O)NC c1(C(=O)NCCC2CCN(C(C(CC)(C)C(N)=O)=O)C2)cccc2nc(C)sc12 Cc1cc(C(N2CCC(CNC(=O)CC3CC34CC4)C2)=O)cc(N)c1 c1(CC(=O)NC2CCC(CNC(C3(C)CSC3)=O)C2)cncc(O)c1 C(=O)(C1CCCc2nnn(C)c21)NCC(=O)NC1(COC)CCN(C(C)=O)C1 N1(C(CCC(C)OCC)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)C(C(C)C)C1 CC1(C)CN(C(=O)C=CC2CCOCC2)CC1NC(C1(c2ccccc2)CC1)=O c1(C(=O)Nc2c(C)cc(F)cc2C)cc2cc(-c3ccnnc3)ccc2s1 C1(C(C)C)CN(C(C2CC2n2cccn2)=O)CCCN1C(=O)C=C1CCC1 c1(CCNC(C(CC2CC2)NC(c2c(C)coc2)=O)=O)ccnc(O)c1 C1(C(=O)NCC2(C)C(C)CN(C(C34CC(CO3)C4)=O)C2)COc2ccccc2O1 C1(C)(CCNC(c2cc(C)c(C)o2)=O)CCN(C(C2CCC(C)(C)O2)=O)CC1 CCCC(C)(C)CC(=O)NCc1cc(C)c(C(N2CCC(C)(F)C2)=O)o1 Cc1nc(C(=O)N(CCCN(C)C(c2cc(F)ccc2O)=O)C)cn(C)c1=O CC12CSCC1CN(C(=O)C(Cn1cncn1)NC(C1CN3CCN1CC3)=O)C2 c1(CSCC(=O)NC2CC2NC(=O)NC2CC(n3ccnn3)C2)ccccc1 C1(NC(CC2C(C)CCCC2)=O)CC2CCC1CN(C(=O)Cc1ccoc1)C2 N1(C(=O)OC(C)(C)C)CC(OC)CC2(CCC2)C1.C12CC3CCCC(C1)N3C(=O)N2 C(=O)(CC(C)(O)COC)N(C1CCN(C(=O)Cn2ncc(Cl)c2C)C1)CC Cc1cccn2nc(C(N3CC(CNC(C4CC4(C)Br)=O)OC(C)(C)C3)=O)cc12 O=C(N=c1ccn(C2CC2(F)F)[nH]1)N1CCCC(Nc2ccc(Cl)cc2)C1 C1(CNC(C2CCN(Cc3cc(C)nn3C)C2)=O)COc2ccccc2O1 c1(C(N2C(CCCNC(C(CCC)CC)=O)CCC2)=O)cnc(C)c(Cl)c1Cl C1(C(C)NC(C2CC(CCC)C2)=O)CN(C(=O)Cc2nc(CC)cs2)CCO1 C1(CCNC(=O)C(c2ccc(F)cn2)(F)F)CCN(C(=O)CCF)CC1(F)F c1(CNC(C(=O)NC(c2noc(-c3ccccc3)n2)C)=O)ncoc1Br C1(C(N2CC(CCC)C(CO)C2)=O)CNC(=O)CN1C(C1CCS(=O)CC1)=O c12cn(nn1)CC(=O)N(C)C2C.C1(CC(=O)NCCO)CCCC1C C(=O)(C1CCc2cccc(F)c21)NCCCCCCNC(c1n(C=C)nnc1)=O C1(NC(COc2c(C)cccc2)=O)CC12CCN(C(C1(C(N)=O)CCC1)=O)CC2 C(C(C)C(F)C(=O)Nc1ncccc1C)NC(C(C)(C)NC(C)=O)=O C1(F)(C(N2CCC(C(C)C)C2)=O)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 C#CC1(C(N2CCC(CC3CC3)C2)=O)CCN(C(c2ncn3ccccc23)=O)C1 c1(C(N2CC3(C(NC(C4CCN(C)C4)=O)CCC3)C2)=O)cc([N+](=O)[O-])cnc1N N1(C(c2cn(C)c(O)n2)=O)CCCC(C2CCCN(C(=O)COC(C)(C)C)C2)C1 c1(CCC(N2CCC(C(=O)NC(c3cnc[nH]3)(C)C)C2)=O)ccccc1Cl Cc1cccc(C(N2CCC3C(NC(C4CCOC4C)=O)C3C2)=O)c1O c1(-n2c(C(C(C)C)OC)nc(-c3ccccc3C)n2)cccc2cnccc12 C1(C(N2CCC(N(C(COCC)=O)C)C2)=O)CC12CCOc1ccccc12 O=C(C1=CCCCCC1)NC1COCC1NC(=O)Cc1ccc(F)cc1Cl CC(C(=O)NCCCCCO)(C1CCC1)NC(=O)CSCCN(C)C CC1CN(C(c2nnn(C)c2C(F)(F)F)=O)CC1NC(c1cc(C(F)F)[nH]n1)=O N1(C(CC=C)=O)CC(C)(C)C(NC(c2ccc(C(C)C)s2)=O)C(C)(C)C1 c1(C(N2CC(C(C(=O)NCC(CC)C#N)O)C2)=O)cc(C)c(C)o1 c1(C(=O)OCC)ccnc(C(N2CCC2CNC(=O)C(Cl)=CCl)=O)c1